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217,C(C(C(=O)NCCC1CN(C(c2cnn(C)n2)=O)C1)OC)OC.n12cc(nn1)C2 218,C(=O)(CC1(NC(=O)NCCOOC)CC1)N(CCC)CC1CC1 219,Cc1cc(CC(=O)NCCC2CN(C(=O)C(C)OCC(C)C)CC2C)ccc1F 220,CC1(C)CC(C)(NC(=O)C(CNC(=O)CCCC2CCCO2)CC2CC2)C1 221,N1(C(CC(C)O)=O)CC2(CNC(c3csc(-c4ncc[nH]4)n3)=O)CC1CO2 222,C1(CCC(=O)NCCCC2CC2)CCCCN1C(c1coc(C(F)F)n1)=O 223,C(=O)(C(CC(C)(C)C)NC(=O)CC(C)(F)F)N(CC(CN(C)C)O)C 224,N1(CC(=O)NCC(CN(C(CCN(CC)CC)=O)C)C)CCCC1=O 225,C(CC(C(=O)N1CCC(OCCC)CC1)NC(C1CCOC1(C)C)=O)=CC 226,c1(CC)ncoc1C(=O)NCCCCNC(C1CSCCS1)=O 227,C(=O)(C(C)(C)CCCN)N1CC(C(=O)OC)C(C(=O)N(C)C)C1 228,C=CCCCC(C(=O)NCCN1CC2CC2C1)NC(C1CCCOCC1)=O 229,c1(C(=O)NC2CC(NC(=O)CCSc3ccccc3)C2)csc2ccccc12 230,CCC(C)(F)C(=O)N1CC(NC(c2cc(-c3ccc(F)cc3)on2)=O)C(C)C1 231,C1(NC(C2C(C=C)OCC2)=O)CC12CCN(C(c1ncoc1CC)=O)CC2 232,C=CC(C)(C)C(=O)NC(CNC(c1ccncc1I)=O)CC 233,C(CCC(=O)NCCOC(=O)N(C)C(c1nc(C)no1)C)OC(C)=O 234,CC(C)C(CC(=O)NC1(C)CCN(C(C2CC3CC3C2)=O)CC1)C(C)C 235,c1(NC(=O)NCCC2CCN(C(C)=O)CC2)ccc(I)nc1Cl 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254,N1(C(C(C)(C)CC#N)=O)CCC(C(=O)NC2CC3CC4C(C3)C24)C(C)(C)C1 255,Cc1cc(F)ccc1C(=O)NCCC(O)CNC(C12CCCC1(C(N)=O)C2)=O 256,c1(CC(=O)N(CCCNC(C2ON=C(C)C2C)=O)C)c[nH]c(=N)nc1O 257,c1(OC)cccc2[nH]c(C(=O)NC3CCN(C(C4C(C(F)F)C4(C)C)=O)C3)cc12 258,C1(CNC(C(=Cc2ccccc2)C)=O)CC2(CC2)CN1C(=O)CC1CC(O)C1(C)C 259,CC(CC1(C)OCCO1)CN=c1[nH]c(=N)[nH]c(=NC2CCCCC2)[nH]1 260,C(=O)(CCCCNC(=O)Cc1cc[nH]c1)N1C(C(=O)OC)C=CC1 261,Cc1ccc(Cl)c(C(=O)Nc2ccc(C(=O)Nc3ncnc(Cl)c3Br)nc2)c1 262,CC(CC(F)(F)F)C(=O)NC1CC(C)(C(=O)N(C2CCCC(C)C2C)C)C1 263,C1(N(C)CC)CCN(C(=O)CCC2(NC(=O)CCCC3CCCO3)CCC2)CC1 264,CCC(CC)(CN=c1[nH]c(OC)ncc1Br)NC(=O)CCOC 265,c1(COc2ccc(NC(CNC(CCOCC)=O)=O)cc2)ccc(Cl)cc1 266,C12C3CC4CN(C1C4C3)C2=O.c1(NC(=O)COC2CCC2)cccc([N+](=O)[O-])c1 267,N1(C(CCC(C)SC)=O)CCC(C2(NC(=O)CC(C)n3ccnc3)CC2)C1 268,c1(OC)ccc(CNC(=O)NCCNCC(O)Cc2ccc(C)cc2)c(Cl)c1 269,N1(C(CCNC(=O)OC)=O)CC=CC1(C)C(=O)NCCc1ccc(O)cn1 270,C(CC(=O)N1CCN(C(C2CC23CC3)=O)CC1)(C(F)F)NC(=O)OC(C)(C)C 271,N1(C(=O)NC2(CCCC)CC2)CCC(N(CC(C2CCCO2)O)C)CC1 272,C(=O)(CCCCCF)NCC(=O)N(CC(C)O)CCCCN(CC)CC 273,C1(CC(=O)NCC(C2CCC2)NC(CC=C(C)C)=O)C(=O)NN=C1C 274,CN1CCC(C(=O)NC2CC(CNC(=O)CC(=O)NC3CC3)C2)C1=O 275,C1(C)(C(=O)NCCC(C(C)C)NC(Cc2ccc(C)o2)=O)CCCNS1(=O)=O 276,c1(C(=O)NCC2C=CC(NC(C(C3CCCC3)OC)=O)C2)ccc(C(C)C)cc1 277,c1(C(N2C(CNC(CSC(C)C)=O)C=CC2)=O)cc([N+](=O)[O-])cc([N+](=O)[O-])c1 278,c1(OC(C)C(N2CCCC(CCCCNC(=O)C(N)=O)C2)=O)ccc(F)c(F)c1 279,C=CC(CC)C(=O)NCC(c1ccccc1F)NC(=O)CNC(=O)CC 280,N1(C(C2(C(=O)OC)CC2)=O)CCCC2CCN(C(=O)C(Br)=C(C)C)CC12 281,c1(C(CNC(Cc2nc(CC)[nH]n2)=O)O)cc(Br)ccc1OC 282,S(=O)(=O)(c1ccc(Cl)c2ncccc12)N1C(CC)C(=O)N(CC)CC1 283,C(CN=C(NCc1cc(Br)ccc1O)NC1CCS(=O)(=O)C1)OCCC 284,CCC(C(=O)NCC(C(=O)NC(C)Cc1ncn(C)n1)C(C)(C)C)C(C)(C)CC 285,N1(C(C2N(C(C)(C)C)CC2)=O)CC2CC(NC(=O)C(F)=C3CCCC3)CC(C2)C1 286,C(=O)(C1=CC2CCCCCC12)NC1(C)CCN(C(=O)CC2CC(=O)C2)C1 287,C(c1cccnc1)=C(C)C(N1CC(CF)(NC(c2cnn(C(C)C)c2)=O)C1)=O 288,c1(C(N2CCC(CC=C)(NC(=O)C(C)COC)C2)=O)ccc(=N)[nH]c1OC 289,CCCC(CCCNC(C1CC(OC)CN1CC)=O)N=c1[nH]c(Cl)nc(C)c1F 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308,CCCC(O)(CNC(c1ccc(NC(=O)CNC)cn1)=O)CCC 309,c1(NC)ccc(C(=O)NCC(C2CCCC2)NC(=O)C(C2CCCCC2)O)nc1 310,CC1(NC(C2CCC(NC(=O)C(O)C3CC3)C2)=O)CC2CCC1C2 311,N(S(=O)(=O)N(C)C)CC(=O)NCC(C1CC1)NC(C(C)N(c1cnccn1)C)=O 312,c1(CC(=O)NC(C2CCCCN2C(c2ncoc2C(C)C)=O)C)ccc(O)nc1 313,N1(CCN(C(=O)C(O)C2CC2)C)CCN(C(=O)CO)CC1.c1cnnn1C 314,S(=O)(=O)(c1ccc(NC(C23CC4CC(CC(C4)C2)C3)C)c(F)c1)NC1CC(C)C1 315,C=CCCCC(C1CC1)NC(=O)NCCc1nccn1-c1ccccc1 316,c1(C(N2CCN(C(=O)CC3CC34CC4)CC2C2CCC2)=O)cncc2c[nH]nc12 317,C1(C)(OC)CCCN(C(=O)Cn2cc(C3(O)COC3)nn2)C1 318,CC1(CNC(=O)CC2CCCO2)CC(F)(F)CN1C(c1ccc(C(F)(F)F)[nH]1)=O 319,c1(C(=O)NCC(CC=C)NC(=O)C(F)C2CCC2)cccc2nccnc12 320,C(=O)(C(=O)C(C)(C)C)N1CCC(NC(C2OCC(C)(C)C2)c2ccccn2)CC1 321,N1(C(C2C(C)(C)COCC2)=O)CCc2[nH]nc(CNC(C3(C)CCOC3)=O)c2C1 322,c1(OC)ccc(F)c(C(N2CCN(C(c3cc(OC)ncc3F)=O)C3CC23)=O)n1 323,O=C(C#CC1CCCCC1)NC(CC(=O)NC(CCO)C(F)F)C1CC1 324,c1(C(=O)NCC(CC)NC(c2ccn(C)c2)=O)cc2cccnc2s1 325,N1(CC(N2C(C)CCCC2C)=O)CC2CC(NC(C3(C)CS(=O)(=O)C3)=O)CC1C2 326,Cc1ncccc1C(=O)NC1CC(CC(=O)Nc2cnccc2C(F)(F)F)C1 327,C1(C(=O)NCc2n(CC)ncc2)CC(NC(=O)CC2CCC(O)C2)CCO1 328,C1(C(C)NC(C2CC(F)(F)C2)=O)CN(C(C2(O)CCOCC2)=O)CCO1 329,N1(C(=O)NCC2COCC(C)(C)O2)CCCC(C)(O)CC1 330,N1(C(c2cc(OC)n[nH]2)=O)CC2CC1(C(=O)NOCCC(C)O)C2 331,c1(C(N2CCC(C(C)NC(C(C(C)C)SC)=O)C2)=O)c(C)nn(CCO)c1C 332,c1(Cn2c(C(C)(CCSC)NCC(COC)(C)C)nnn2)nn(C)c(Cl)c1Br 333,Fc1ccc(C2=CCN(CC(c3ccccc3)Nc3ccco3)CC2)cc1 334,c1(C(=O)NCC=CCNC(CCn2ccc(C)n2)=O)cc2c(s1)CCCNC2=O 335,N1(C(CCC=CC)=O)CC2CCC1CN2C(=O)CSc1ccccc1C 336,c1(N(C)C)ccc(C=CC(N2CCC(NC(=O)C(F)C3CC3)C(O)C2)=O)cc1 337,CC(C(=O)OC(C)(C)C)C(=O)NC1CN(C(c2ccc[n+]([O-])c2)=O)CC1C 338,c1(NC(c2cc(Cl)no2)C)[nH]c(=NCC2CCN(C)C(=O)C2)nc2c1cnn2C 339,C=C(C)CCC(=O)N1CCC(CNC(=O)C(C)OCC(F)(F)F)C1 340,CC1(C)CC(C(N2CC(NC(=O)Cc3c[nH]nc3O)C(O)C2)=O)CC(C)(C)S1 341,c1(CNC(C2C3CCC23)=O)cnn2c1CN(C(C1CCCC13OCCO3)=O)CC2 342,c1(SC)ccc([N+](=O)[O-])c(C(N2CC3CC(NC(=O)C(C)(C)C)CC3C2)=O)c1 343,c1(C(N2CCC(N(C(=O)C(O)CC(F)F)CCO)C2)=O)cc2c(s1)CCC2 344,c1(C(N(CC(C)NC(C(CC=C)c2ccccc2)=O)C)=O)csc([N+](=O)[O-])c1 345,c1(C(c2n(CCC)nnn2)NC2COC2)cn(C)nc1-c1ccccc1 346,N1(C(c2cc(CC)on2)=O)CCN(C(=O)COCC(=O)OC)C(CF)C1 347,N1(C(c2nnc(CC)s2)=O)CCCC(C2CC2NC(C2CCCS2)=O)C1 348,C1(CCC)CCCN(C(c2csc(CNC(=O)Cc3cnc(C)s3)c2)=O)CC1 349,c1(C(N2C3CC(NC(C(C=C)O)=O)CC2CC3)=O)csc2ccc(Br)cc12 350,Cc1ccc(C(=O)NC(CNC(c2ccc(C#N)s2)=O)CO)c(=O)n1C 351,C#Cc1ccccc1CNC(=O)C(C)(C)NC(c1ccn(C(F)F)n1)=O 352,N1(C(C(C)NC(=O)OC)=O)CCC2(C1)CN(C(=O)Cc1ccccc1C)CCO2 353,C12(CC(=O)NC(CCNC(c3cnc(C)n3C)=O)C)CC3CC(CC(C3)C1)C2 354,C1(C(C)(C)NC(CSCC(C)C)=O)CCCN1C(=O)Cc1cc(C2CC2)n[nH]1 355,N1(C(CC(CCC)O)=O)CCc2nc(CNC(c3csc4nnsc34)=O)sc2C1 356,C1(C(N2CC(C)(CCC(=O)NCCCC3CCOCC3)C2)=O)CCS(=O)(=O)C1 357,C(=O)(CCCC1CC1)NC(c1ccccc1)C(=O)N(CC(C)(C)OC)C 358,CCCC(C(=O)NCc1ccc(-n2cc(CCCO)nn2)cc1)S(N)(=O)=O 359,CCCC(C(=O)OC)C(=O)NC12CC(CNC(=O)Cc3coc(C)n3)(C1)C2 360,CC1(C(N2CC(C#N)C2)=O)CN(C(=O)CNC(=O)C(C)(C)C)C1 361,CC1(C(=O)O)CN(C(c2cc(C(=O)O)nn2C2CCCC2)=O)CCO1 362,c1(OC)ccc(F)cc1CC(=O)N(CCCN(C(=O)C1=CCCCC1)C)C 363,c1(OC)cncc(C(=O)N(C)CC2CCCN2C(c2ccnn2C(F)F)=O)c1C 364,C(=O)(C1=C(Cl)CCOC1)NCc1cn(CC(=O)NC(c2ccccc2)C)nn1 365,C(=O)(CC(C)CC(=O)OC)N1CC2C(CC(=O)NC3(CC=C)CCC3)C2C1 366,C(CN=c1[nH]c(=NCC2CCC(=O)NC2)[nH]c2c1CSC2)SCC 367,c1(CC(N2CCC(NC(CCC3C(C)C3)=O)C2C)=O)c[nH]c2cnccc12 368,C(=O)(C(O)CNC(c1sccc1CO)=O)N(CCOCCOC)C 369,C1(C(=O)NCC=C(C)C)C2CC(O)C(C2)N1C(C1CS(=O)(=O)C1)=O 370,CCCCCCCCCC(C)CC(=O)NCCCNC(c1ccnc(Cl)c1O)=O 371,C(=O)(C(CN(C)C)C(C)C)N1C(CNC(CC2(OC)CCC2)=O)CC1 372,N1(CC)CCCC(c2cn(CC(N3CCCN(CC(N)=O)CC3)=O)nn2)C1=O 373,N1(C(C(C2CCOC2)OC)=O)CCC(C)C(CNC(=O)C=CC2CC2)C1 374,O=C1NCC2CCCN(C(c3cncnc3)C(=O)NC3CCOC3)C12 375,N1(C(C(CC(C)C)N(C)C(c2cccc(O)c2F)=O)=O)CCN2C(=O)OCC2C1 376,c1(NCC)cccc(C(=O)NCC2CC2NC(C2CCNC2=O)=O)c1 377,C(=O)(C1=NOC(C)C1)N(CC)CC1CCCN1C(=O)Cc1csc(Br)c1 378,Cc1onc(Br)c1CNC(c1nnnn1C1CCCC1)C1CCC1.c1cn(C)cn1 379,c1(OC)cccc2c(C(N3CCN(C(=O)C(Cl)=CCl)CC3C(C)C)=O)cccc12 380,C(=O)(CCCCCF)NCc1c(C(N(C(C)C(C)(C)O)C)=O)nco1 381,C1(C(=O)NCc2nncs2)CCN(C(C2(CCF)CCC2)=O)CCO1 382,N1(c2nnc(C(N)=O)s2)CCOCC(CNC(=O)C(C2CC2)C2CC2)C1 383,C(=O)(C1Cc2cccc(Br)c21)NC1CCC(NC(C(C)C)=O)C1 384,c1(C(N2CCN(C(C3CCCS3)=O)C3C2CCC3)=O)cc(=O)c2ccccc2o1 385,N1(C(c2c(C)nc(C3CC3)s2)=O)CCN(C(=O)CC2(O)CCC2)CC1C(C)C 386,C1(NC(C(C2CC(F)(F)C2)OC)=O)CCN(C(c2ccc(C)nc2N)=O)C1(C)C 387,N1(C(C(COC)C)=O)CC(CC(=O)NCCc2cnccn2)C(C)C1 388,c1(C(C)C)c(C(N2CCCC2C(C)NC(C2CCC(=O)N2)=O)=O)cccc1F 389,c1(OCC(=O)NC2CC(C)(NC(Cn3ccc(C)n3)=O)C2)ccc(F)cc1Cl 390,n1(C(C)C)cnc2c(N(C)CCF)nc(N3CCC(C(F)(F)F)C(C)C3)nc12 391,C1(NC(Cn2c(C(C)C)ncc2)=O)CN(C(=O)CCC2(C)CC2)C2(CCCC2)C1 392,CC(CN(C)C(C1(N(C)C)CCC1)=O)C(=O)NCCc1cscn1 393,N1(C(C(C(CC)C)O)=O)CCC2(CCC(CNC(c3ccc[nH]3)=O)CC2)CC1 394,C1(C)(CC)CC(NC(=O)CCN(C)C(C)=O)CN1C(c1cnn(C(C)C)c1F)=O 395,CCC(CC(=O)NC1CC(C)(NC(=O)COCC(=O)Nc2nc[nH]n2)C1)SC 396,n1(CC(=O)NC(c2scc(C(=O)OCC)n2)C)c(S)nc2ccccc2c1=O 397,CC(CNC(=O)OC(C)(C)C)CC(=O)N1CCC1CNC(C1(CO)CC1)=O 398,C1(F)(CNC(c2noc(CC)c2C)=O)CCCN(C(C2CC2c2nc[nH]n2)=O)CC1 399,C=C(Cl)CC(C(=O)NC(c1cc[nH]n1)C)NC(c1cnc(O)cc1C)=O 400,c1(C(C(=O)NC2C(CNC(C3(C=C)CCC3)=O)CC2)O)cc(F)c(F)c(F)c1 401,C1(CC(=O)NC(C(=O)OC)C)CC(C)(C)CN1C(C1CCC(OC)CC1)=O 402,CC(CCN(CCCN1CCNCC1)C)CC(C)(C)C 403,C1(NC(c2nc(N(C)C)oc2)=O)CCSC12CN(C(=O)CC=C(Cl)Cl)C2 404,c1(CSc2c(C)nn(-c3cccc(Br)c3)c2Cl)cn(-c2ccccc2)c(=O)nc1O 405,C(=O)(C1CCCc2ncnn21)NC1C(OC)CN(C(c2cncc(C#C)c2)=O)C1 406,n1(-c2ccn(CC)n2)nc(CCCc2ccccc2)nc1CCc1ccccn1 407,N1(C(c2c(N)ccc(F)c2)=O)CCN(C(c2cc(O)ncn2)=O)C2CCCCC12 408,C(=O)(C(C)(F)C(=O)OC)N1CCC(CCC)C1.C(=O)(CCN1CCCC1)N 409,CCCCC(O)C(C)C(=O)NCC1(O)CCN(C(=O)C=Cc2ccncn2)CC1 410,CN1N=C(CC(=O)N2CCC(F)(F)C(CNC(C3(O)CCSCC3)=O)C2)CC1=O 411,c1(C(=O)NC2C3CCN(C(CCCCC=C)=O)C32)cccc2c1OC(C)(C)C2 412,C1(OC(C)(C)C)CC(C(N)=O)C(NC(=O)NC2C3CC3C3CC23)C1 413,CCCCC(C(=O)NCCc1cccc(O)n1)NC(=O)CCc1cnoc1 414,N1(C(C2(CC#C)CN(C(=O)OC(C)(C)C)CCO2)=O)CCC(F)(F)CC(C)C1 415,c1(CCC)c(C(=O)NC2(CO)CCN(C(c3cccnn3)=O)C2)nnn1C 416,CCCC(C(=O)NCC1CCCCN1CCOc1cccc(Cl)c1)OC 417,CC(C(=O)OC(C)(C)C)C(=O)N1CCC(C(C)NC(=O)CCc2cnc(O)[nH]2)C1 418,Cn1cnc(CC(=O)NCC2C=CCN2C(=O)CCc2nnc(C(F)F)o2)c1 419,C1(C(=O)NCCN(CCOC)C(c2cc(COC(C)(C)C)on2)=O)CC=CCC1C 420,N(C1CCc2ccccc21)C(C(CNC(c1ncnc(C)c1C)=O)O)=O 421,C12(C(N3CCC(CNC(CC(C)N(C)C)=O)C3)=O)CCC(CC1)OC2 422,C(=O)(C1CCc2cccc(Cl)c21)N1C2CC(NC(C3(CC)COC3)=O)CC1CC2 423,C1(C(=O)NCCOC2CN(C(c3ccc(=N)[nH]c3)=O)C2)CC2(CCOCC2)CO1 424,C1(NC(c2c(C)cc(SC)s2)=O)CCCC12CN(C(=O)CCC#N)C2 425,c1(NCC2(CNC(=O)Cc3cnns3)CCCC2)cc(C(=O)O)ccc1[N+](=O)[O-] 426,S(=O)(=O)(c1cccnc1)N1CCC(C(N2CC(F)CC(C(=O)OC)C2)=O)CC1 427,c1(Sc2n(C)nnn2)cc(F)cc(F)c1Oc1cccc(F)c1 428,N1(C(CS(CC)=O)=O)CC2CCCC2(NC(C23CC(COC)(CO2)C3)=O)C1 429,C1(NC(c2c(C)cno2)=O)C=CCN(C(=O)Cn2cccc2)C1 430,O=C1NC(C(=O)NCC2CCN2C(=O)Cn2cnccc2=O)CCO1 431,C(Cc1ccoc1)(C(=O)NOCCF)NC(C1CCCC(=O)C1)=O 432,c1(C(C)OC(=O)NC(CC(=O)NC)C)ccc(Cl)c(Cl)c1 433,c1(C(N2CCCC(NC(c3c(C)[nH]cc3)=O)C2)=O)cn(C)c(=O)cn1 434,C1(C(N2C(CCNC(C3N(C)CC(F)C3)=O)CCCC2)=O)CC(C)(C)OC1=O 435,C(N=C(NC1CCCC1)N1CC(O)C2(CC2)C1)C1C(C)(C)C2CCC1C2 436,N1(C(CCOCCC)=O)CCCC2CCN(C(c3cccn4cncc34)=O)CC12 437,N1(C(c2c(CCC)nco2)=O)CCC2(CC1)CC2C(=O)NC1(C)CCCC1(C)C 438,c1(C(=O)NCC(CNC(C(C)Cc2cnn(C)c2)=O)(C)O)cc2n(c1)CCOC2 439,C1(NC(n2ncnn2)=O)CN(C(=O)COCCOCCO)CC(F)(F)C1 440,C1(NC(C(C)SCC)=O)CCCCC1CNC(c1ccn(C)c1CC)=O 441,N1(C(CCCC2(C)N=N2)=O)CC(NC(c2cc(C3CC3)on2)=O)C2CCCCC12 442,c1(NC(CCC(C)(C)C)c2nnnn2CC2CC2)ccc2c(c1)C(=O)NCCC2 443,c1(CNC2C(C)CN(C(N3CCOCC(C)(CO)C3)=O)C2)cccc2c[nH]nc12 444,c1(NC(c2nnnn2CCCC2CC2)CCC)cc([N+](=O)[O-])ccc1C 445,CCCC(C(=O)N1CCCCC12CC(NC(=O)C(C)(CC)CC)C2)S(N)(=O)=O 446,C1(NC(C(n2cc(-c3c(OC)nc(C)cc3)nn2)C)=O)CCOC2(CCSC2)C1 447,c1(COC)cccc2sc(NC(c3sc(C(F)(F)F)cc3Br)=O)nc12 448,c1(NC(C23C(CN(C(C(C)OC4CC4)=O)C2)CC3)=O)ccc2c(c1)OCO2 449,c1(C(=O)NC2C(CNC(c3cc(Cl)no3)=O)COC2)coc2ccc(Cl)cc12 450,CC(C)C(CO)C(=O)NCC(C)CNC(=O)CC1CC2CCC1C2 451,C(=O)(C(CO)C(C)(C)C)N1C(CN(C(Cc2nc(C(C)OC)sc2)=O)C)CCC1 452,CCC(CO)C(=O)N1CC(CN(C)C(c2c(OC)noc2C)=O)C1 453,C12(C(N(CC(N3CCCC(CO)C3)=O)CC)=O)CCC(CC1=O)C2 454,CCCC(C)(O)CC(=O)N(C)CCOCCN(c1nnccc1C#N)C 455,c1(C(=O)NCC2CCCC(NC(CCC(=C)C)=O)C2)ccc2c(=O)cc[nH]c2c1 456,C1(NC(C(C2(O)CN(C(c3csc(C)c3C)=O)C2)F)=O)CCCCCC1O 457,N1(C(C(C2CCOCC2)C)=O)CC(N(C)C(c2c[nH]nc2Br)=O)C(C)(C)C1 458,CC(C)C(C)C(=O)N1CC2C(CNC(=O)CCOCc3ccccc3)C2C1 459,Cc1ccc([N+](=O)[O-])c(NNC(=O)NCC23CNCC2(C)C3)n1 460,C1(C(=O)NC2CCN(C(Cc3nc(C(C)(C)C)sc3)=O)C2)CC2(CCC2)CCO1 461,c1(C(=O)OC)cnc(NC(C2CC(F)CN(C(C3(C)COC3)=O)C2)=O)c(I)c1 462,N1(C(CC(=O)OC)=O)CC(C2CN(C(c3cccc(-c4nnc(C)o4)c3)=O)C2)C1 463,N1(C(C=CC=CC)=O)CC(C)CN(C(c2ccc(SC)cc2OC)=O)C(C)C1 464,c1(C(=O)NCCC(C)CCNC(=O)C(F)CC2CC2)cccc2ccnn12 465,C(N=c1[nH]c(=NC2CC=CCC2C(F)(F)F)[nH]c2c1COC2)C1(CCC)CCC1 466,Cc1c(C(N2CCOC(CN(C)C)C2)=O)cnn1CCC(C)C 467,N1(C(C(CC)=CCCC)=O)CC(C)CN(C(c2ccc(C(F)F)cc2)=O)CC1C 468,C1(C(=O)NC(c2ccccc2F)C)CC(F)CN1C(=O)C(c1ccccc1)O 469,N1(C(CCCn2ncc(C)c2)=O)CCC(n2cc(CNC=O)nn2)CC1 470,N1(C(C(c2cccc(OC)c2)(F)F)=O)CC(NC(c2nncs2)=O)CC(O)C1 471,C=C(Cl)CCC(=O)NCC(C)(CNC(c1csc(C(C)=O)n1)=O)OC 472,c1(Cn2cc(-c3scc(-c4cccc(F)c4)n3)nn2)cccc2ccccc12 473,C1(CC=C)(NC(CCN(C(=O)C(O)CN(C)C)CC#C)=O)CCCC1 474,c1(-c2cn(CCC3N(C(CC(C)F)=O)CCSC3)nn2)c2c(nn1C)CCCC2 475,C=CC1CN(C(c2ccc(F)c(O)c2)=O)CC1NC(C1CCC(F)(F)CO1)=O 476,N1(C(CCC#N)=O)CCC(CNC(c2cccc3nccn23)=O)C(F)(F)C1 477,c1(C(=O)NCC(C2CC2)NC(c2cnc(CC)s2)=O)c(F)cncc1Cl 478,c1(C(=O)NCC2(F)CC(NC(C(CC=C)(C)C)=O)C2)cc(F)c(C#N)c(F)c1 479,C1(NC(c2c(C)oc(-c3cnn(C)c3)n2)=O)CCCCN(C(=O)C2=CCCC2)C1 480,c1(C(=O)NOCc2cn(CC3(O)CC3)nn2)ccc(C(F)(F)F)cn1 481,C1(NC(C(C)N2CCCC2)=O)CCN(C(C2CC3(CC(=O)C3)C2)=O)C1(C)C 482,C1(CNC(c2c(SCC)cncc2)=O)COCCN(C(C2(C)CCCN2C)=O)C1 483,C1(CNC(C(C)N2CCC2)=O)CC2CCC1N(C(=O)CC(C)c1cccnc1)C2 484,c1(OC)ccc(Cl)cc1C(N1CCN(Cc2cn(C3C=CCCC3)nn2)CC1)=O 485,Cc1c(NCc2cnc(O)nc2O)ncnc1NC(c1cccnc1)C 486,C(C)(CCCCNC(=O)C(C)(O)C1CCC1)NC(CC1(C=C)CCC1)=O 487,Cn1ccc2cccc(C(N3CC(F)CC3C(=O)Nc3cccc(N)c3)=O)c12 488,C(=O)(CCCCC(=O)NC1CC(OC)CN(C(c2coc(N(C)C)n2)=O)C1)OC 489,C(=O)(C(O)C(C)CC)NC(CC=C)CNC(c1ccc(C(N)=O)cc1)=O 490,c1(N2CCCC(NC(CCCN(CCC)CCC)=O)C2C)nc2ncc(Cl)cc2s1 491,C1(C(=O)OCC(C)(C)OCCCCCC)CCS(=O)(=O)CN1C(C)=O 492,C(=O)(C1CCc2c[nH]nc21)N(C(C(=O)NC1C(C)CCCCC1)C1CC1)C 493,C1(NC(C=CCC)=O)CC2CCC1CN2C(=O)Cn1cc(C2CC2)cn1 494,C#Cc1cc(NC(=O)CN(C(=O)C(C(C)CC)N(C)C)CC(C)(C)C)cc(F)c1 495,N1(C(C2C=CC(NC(C#CC(C)(C)O)=O)C2)=O)CCOC2(CCCC2)C1 496,N#CC1CCCCN1C(C1CN(C(c2cccc(C(F)(F)F)c2)=O)C1)=O 497,C(c1ccnn1C)=CC(=O)NCC1(CNC(C(N2CCCCC2)C)=O)CCCC1 498,C1(C(=O)OC(CC)C(=O)N(C)CC)CCN(c2ccc(CC(C)C)nc2)CC1 499,c1(C(N(CCCNC(Cc2c(CC)con2)=O)C)=O)cn(C2CC2)c(C)cc1=O 500,N1(C(C(CC)C)=O)CCC(C(C)NC(C2CC23CCOC3)=O)CC1 501,c1(C(=O)NC2C(NC(C(F)=CC)=O)CCCC2)cn2c(Br)cnc2s1 502,C(=O)(CCCC(N)=O)NCCC1C(C)CN(C(c2c[nH]nc2Br)=O)C1 503,CC(O)(CC(=O)N1CC=CC(NC(=O)CCCCN2CCCC2)C1)C(F)(F)F 504,N1(C(C(C)N(C)C)=O)CCC2(CCC(NC(c3cnc(O)o3)=O)C2)C1 505,CC(CNC(c1ccnnc1)=O)CC(=O)N(C1CCCC1)C 506,n1(CC)cc(Br)c(C2CCCN2C(=O)CNc2cnn(C)c2)n1 507,C1(c2ccc(Cl)cc2)(C(=O)NCCCN(C(COC)=O)C2CC2)CCN(C)C1 508,N1(C(CSCCC)=O)CCCCC(C2CN(C(=O)Cc3ccccc3C)C2)C1 509,c1(C(=O)NC(COC)CNC(C2CCC3CC23)=O)ccc(C2CC2)c(F)c1 510,Cn1ncc2c1CCC(C(N1C3CCCC1CN(C(=O)CC(C)(C)O)C3)=O)C2 511,c1(C(N2C(CNC(C3(F)C(C)C3)=O)CC2)=O)cc2cc(Cl)ccc2o1 512,C1(NC(C(C(C)C)(C)C)=O)CCCN(C(=O)CC(F)F)CC1F 513,CC1CCCC1(C(=O)NC(C(O)CO)C1CC1)NC(c1cnn(C2CC2)c1)=O 514,CC(C)(C(=O)NC1CC1CNC(=O)CCN1CCCC1=O)N1CCCCC1 515,CCN=c1[nH]cc(C(=O)NC(C)(CNC(C2CCCN2CC)=O)CO)s1 516,C(=O)(C(CC)C(=O)NC(c1cccnc1)C(=O)NCCOC1CCCC1)OCC 517,c1(C(=O)NCCCN(CCCNC(C(CC)N(C)C)=O)C)cnc2[nH]cnc2c1 518,c1(OC)ccc(CCC(=O)NCCNC(=O)CC2COCCOC2)cc1N 519,N1(C(C(C)C(C)(C)C)=O)CCCN(C(c2cncc(C3CC3)c2)=O)CC1C 520,CC1CCC(CCC(=O)NCC(C)(C)CNC(C23CC(CC(F)F)(C2)C3)=O)O1 521,c1(C(=O)NCC2(CCNC(c3n(C)ncc3)=O)CC2)cc(N2CCCC2)ccn1 522,N1(C(C)=O)CC2CC1C2C(=O)NC1(c2nn(-c3ccccc3)cc2C)COC1 523,C1(NC(C2CCCN(CC)C2)=O)CCN(C(C2CCCC2C(C)C)=O)C12CCC2 524,N1(C(c2c(=N)cc[nH]c2)=O)CCC2(CCCN(C(C34CCC(CC3)C4)=O)C2)CC1 525,c1(C(=O)NCCC2CCC(NC(C=CC(=O)OCC)=O)C2)n[nH]c2c1COCC2 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599,N1(C(C2(C#C)CC2)=O)CCC(NC(c2c[nH]cc2-c2ccc(C)s2)=O)C(C)C1 600,N1(C(C(CN(C)C)O)=O)CC(NC(=O)CSCc2cccs2)C(C)(C)C1 601,C12(CNC(C(CCSC)(C)C)=O)CC(C(N)=O)(C1)C1(CN(C(=O)C(C)(F)F)C1)O2 602,c1(CC(=O)NCC2(CNC(COCC(=C)C)=O)COC2)cc(F)ccc1F 603,N1(C(c2cscc2F)=O)CCN(C(c2cccc(F)c2Cl)=O)C2COCC12 604,CC1(C(=O)NC2CCCN(C(=O)C3=CS(=O)CCC3)CC2)Cc2ccccc2C1 605,C12CCCC(C1)NC2=O.c1(CN(C(=O)C(=O)OCC(N)=O)CCl)ccc(OC)cc1 606,c1(CCCC(N2CCC(CN(C(C3C(C)C3C)=O)C)C2)=O)nc2ccccc2[nH]1 607,c1(C(N2CCCC(N(C)C(C3CC34CCC4)=O)CC2)=O)ccc2c(c1)CCCS2 608,C=C(C)CC(C)C(=O)NCC(=O)NOCC(F)(F)F 609,C1(NC(CC(=O)OC(C)(C)C)=O)CC2(NC(C3CC4CCC3CC4)=O)COC1C2 610,C#CC1CCCN(C(=O)COC(C)(C)CNC(=O)CC(C)C(F)F)CC1 611,Cc1cc(C(=O)NCc2cn(Cc3ccc(F)c(F)c3)nn2)ccc1S(N)(=O)=O 612,C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NC1CN(C(c2cc(Cl)cnn2)=O)C1 613,C(=O)(C(C(C)(C)O)NC(=O)CC1CC2(CC2)CO1)NCCC(CC)(F)F 614,C1(F)(C(N(CCC(C)NC(C2CCCC23CC3)=O)C)=O)CCC(F)(F)CC1 615,C1(CNC(CC2(C(=C)F)CCC2)=O)CCCCCN1C(=O)C=Cc1cc[nH]c1 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634,C1(COC)CN(C(c2ccc(Cl)cn2)=O)CCN1C(c1ccc(F)c(CO)c1)=O 635,CCC(CC)C(=O)N1CC=CC1(C(=O)NC1C(C)C1(C)C)COC 636,c1(OC)ccc(OC)c(CCC(=O)NC(C)CN(C(=O)C(C)C2CCCO2)C)c1 637,N1(C(C2(CC)CCN(C(=O)CC(C)C(F)F)CC2)=O)CC2(COC(=O)C2)C1 638,C1(C)(CSC)CCN(C(C2(OC)CN(C(C3COCC3(C)C)=O)C2)=O)CC1 639,C(=O)(C(C)C(C)(C)c1ccccc1)NC1CCC(NC(c2ccc(SC)s2)=O)CC1 640,N1(C(C(CC#C)C)=O)CC(NC(=O)C(C2CC2)C2CC2)CCC(O)C1 641,Cc1nn(C)cc1S(=O)(=O)N1CC2C(C(=O)NC(CO)C(C)C)C2C1 642,Cc1ccc(C(N2CCCC(NC(c3ccn(C)n3)=O)C2C)=O)c(F)c1Cl 643,c1(C(N2CCC(NC(C(C=CC)O)=O)C(O)C2)=O)ccc2c(C)[nH]nc2c1 644,C(=O)(CC(CC)C1CC1)NCC(CNC(C(C)(C)OCCC)=O)(C)F 645,C1(CNC(=O)CN2CCCC2)CN(C(C2CC3CCC(C2)C3O)=O)C2(CCC2)C1 646,C(=O)(C1=CC2CC(C1)CC2O)NCC1N(C(CCC(=O)NCCC)=O)CCC1 647,C1(C(N2CCC(CCNC(C3(N(C)C)CCCSC3)=O)C2)=O)OCCCC1(C)C 648,N1(C(C2(CC(C)C)COC2)=O)CC2OCCN(C(=O)C(F)CC(C)C)C2C1 649,C(=O)(C(C(=O)N1CCC(CNC(C2(C(F)(F)F)CC2)=O)C1(C)C)C(C)C)OCC 650,C1(NC(c2c(CC)nns2)=O)(CO)CCN(C(C2(OC)CC(CF)C2)=O)C1 651,Cc1cc(N(C)C(C2CSC(c3ccc(C(F)(F)F)cc3)C2)=O)cc(F)c1 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707,c1(CSC)cc(C(=O)NC2CN(C(c3cc(C)c(Cl)cn3)=O)CC2F)ccc1F 708,CC1CC(NC(c2ccc(C(F)F)cc2)=O)CN1C(=O)C(F)=CC1CC1 709,c1(C(N2CCC(CCCNC(C3CCCC3)=O)CC2)=O)c(O)cc(F)cc1F 710,N1(C(C2CC(OC)C2)=O)CCC2(CCC2)C(NC(=O)C(n2nc(C)cc2C)C)C1 711,c1(C(c2n(CC)nnn2)NC2CC=CCC2)ccc(-c2ccnn2C)cc1.C1(C)CC1 712,c1(NC(C(C)NC(c2ccc(CO)nc2)=O)=O)cccc2ccoc12 713,C(=O)(C(O)C1=CCCCC1)NCCCCCCC(=O)NCCC1CCC(C)CC1 714,N12CCN(CC1)C1CCN(CC1)C2=O.C(CCCOCC(F)(F)F)OC(C)(C)C 715,c1(C(=O)NC(C(C)NC(C2COCCO2)=O)(C)C)ccc2cn(C)nc2c1 716,Cc1ncc(Cl)cc1NC(C1CCC(C2CC2)N1C(=O)Cc1cccn1C)=O 717,N1(C(C(CCCC)O)=O)CC2CCCC(C1)N2C(c1[nH]c(=N)ccc1C)=O 718,C1(CC(C)NC(=O)CCCn2cc(C(C)(C)C(=O)O)nn2)COCCO1 719,O=S(=O)(c1c[nH]c2ncccc12)NCCc1nc(-c2cccs2)n[nH]1 720,C1(NC(C(C)Sc2ccccn2)=O)CCCC12CN(C(=O)Cn1cnnc1)C2 721,N1(C(c2cc(C)c(C)o2)=O)CCC(C(=O)NCc2cc(Cl)no2)C(C)(C)C1 722,N1(C(C2=C(C)OCCS2)=O)CC(C)OC2(CCN(C(c3ccc(=N)[nH]n3)=O)C2)C1 723,O=C(C(O)CC(F)F)NCc1cc(Cl)cnc1Cl 724,N1(c2ccnc3c2COCC3)CCC2CCCCCC2C1 725,O=C(CC(C(F)F)n1cccn1)N1CCCC(C(N2CCCC2)=O)CC1 726,c1(NC(C)=O)ncc(S(=O)(=O)N2CCC(C(=O)NCC(N3CCCCC3)C)CC2)s1 727,C=C(C)CC(C(=O)N1CC(C(N)=O)C2(CC2)C1)NC(c1sccc1C#N)=O 728,C1(C(C)NC(c2cccs2)=O)CN(C(c2c[nH]nc2Br)=O)CCO1 729,c1(C(=O)NC2C3(CC(NC(C(C)CN4CCCCC4)=O)C3)C2)cccc(N)c1F 730,C1(CC(=O)NCC2COCC(C)O2)C2CCCC2N1C(C1CCC1C#N)=O 731,C1(C(=O)NCC(C)NC(=O)CN2CC(C)(C)C2)COc2ccc(O)cc2O1 732,C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)N1CC(NC(C=C(CC)C)=O)C(C)CC1 733,C1(C(=O)OC)CCCC(C(=O)NC23CC(CNC(=O)C(C)C4CCOC4)(C2)C3)C1 734,N1(C(C2N(C(c3ccc(CC)[nH]3)=O)C(C)C2)=O)CCn2cc(C)nc2C1 735,C1(N(C)C)CCCC(N=c2[nH]c(=NCc3ccnc(O)c3)[nH]c3c2COCC3)C1 736,CC(C)CC(C(=O)NCC(C)NC(=O)N)N(C)C.c1(C(=O)NCCSC)cccnn1 737,C1(C(=O)NCc2scc(C(N)=O)n2)CC=CCN1C(=O)CCc1nncs1 738,N1(C(c2cn(C(C)C)nc2)=O)CCN(C(=O)COc2ccc(F)cc2)C(C)C1C 739,C1(CNC(c2c(CC)nc[nH]2)=O)CN(C)CCN1C(=O)COc1ccsn1 740,C(=O)(C#CC1CCCCO1)NC1(C)CCN(C(Cn2nc(C)oc2=O)=O)CC1 741,S(=O)(=O)(c1cc(NC(=O)OC(C)(C)C)ccc1Cl)N(C1CC(C)N(C)CC1)C 742,CCC(C(=O)NCCCC(C)NC(c1ccc(C)nc1N)=O)C(C)C 743,C1(CC(=O)NCCCNC(C2(OCC)CCCC2)=O)CC(OC)C1(C)C 744,N1(C(CCC#C)=O)CCC(=O)NC2CN(C(=O)CCCC(F)(F)F)CCC12 745,C1(CNC(=O)NCC(C)OC)CN(c2cc(C3CC3)ncn2)CCO1 746,Cc1ccc(=N)[nH]c1C(N1CCN(C(=O)C(C)C2CCCC2)CC1C)=O 747,C1(C(C)NC(C(F)OC)=O)CCN(C(c2ccccc2OCF)=O)CC1 748,C1(C)(NC(CC2CCCN(C(C(C)NC(CC)=O)=O)CC2)=O)CCC2(CC1)CC2 749,N1(C(c2cc(CC)oc2C)=O)C2CCC(C2)C1C(=O)NC1CCNC(=O)C1 750,c1(NC(C2CCN(C(CC3(C=C)CC3)=O)C2C)=O)ccc(OCC)c(Cl)c1 751,c1(OCC)nc(N(CCCN(C(=O)C(CO)c2ccccc2)C)C)ncc1Cl 752,C1(C(=O)N(C2CCC(NC(=O)C(C)NC=O)CC2)C)(OC)CCCCC1 753,N1(C(c2c(C)nncc2)=O)CCC(n2cccn2)(CNC(C2CCSCC2)=O)CC1 754,N1(C(C(OC)OC)=O)CC(CO)C2(C1)CN(C(=O)C(CC(C)C)NC(C)=O)C2 755,Cc1cccc(CNC(C23CC2CN(C(C2CCC(=O)N2C)=O)C3)=O)c1O 756,c1(NCC=CCNC(Cc2cc(CC)on2)=O)cc(=O)n2cc(Cl)ccc2n1 757,n1(CC)ccnc1C=CC(N1CCC1CNC(=O)Cc1ccc(C)o1)=O 758,C1(C(=O)NCCCN(C(=O)Cc2cncc(O)c2)CC)CCCCN1C 759,C#CCC(C)(C(=O)NC(c1cnc[nH]1)C)NC(C1CCCC(=O)CC1)=O 760,c1(N2C(C(=O)NCc3cn(C(C)C)nc3)CC(F)C2)ncnc2c(Br)csc12 761,C1(C(N(C)CC2(O)CCN(C(COC(C)=O)=O)C2)=O)CCc2ccnn2C1 762,C1(CNC(C(=O)NCCc2nc(-c3ccc(C)o3)sc2)=O)COCC(C)O1 763,C(=O)(CCCCCC(C)(C)C)NCC1(OC)CCN(C(CC=C=C)=O)C1 764,N1(C(C=C(C)C)=O)CCCC2(CCN(C(c3c(Cl)ccc(Cl)c3O)=O)CC2)C1 765,C1(NC(CCC(C)N(C)C)=O)CC2(C1)CC(NC(C1CCC1C)=O)C2 766,Cc1cc(C(=O)NC2CCC2CNC(c2cn(CC(F)(F)F)nn2)=O)n[nH]1 767,c1(CC(=O)NCC(CN(C(C(C2CCCC2)OC)=O)C)O)cccc2occc12 768,C(=O)(C1=CCCCCC1)NC1C(N(C)C(C2CC23CCOCC3)=O)CCCC1 769,C1(C)(C(=O)NCC2CCCC(NC(COCC#C)=O)C2)CCOC(C)C1 770,C1(C2CCCN(C(=O)Cn3nc(C)ccc3=O)C2)(NC(C2CC(OC)C2)=O)CC1 771,c1(NC)c(C(=O)NC(C)CNC(=O)CC2CC3CC3C2)cccc1[N+](=O)[O-] 772,Cc1cnn(CC(=O)N(C)CC2(O)CN(C(c3cc(C(N)=O)cs3)=O)C2)c1 773,C(=O)(CCS(=O)(=O)c1ccc(Cl)cc1)NC(C(C)NC(CC(C)OC)=O)C 774,N1(C(c2c(CC)nccn2)=O)CCC2(CC1)CCN2C(=O)CCC1CCOC1 775,C1(C(N(C(=O)C=CC(C)(C)C)C)C2CC2)CCN(C(C2CC(N(C)C)C2)=O)C1 776,c1(C(=O)NCCCN(C(c2cncc(OC)n2)=O)C(C)C)cnc(O)c(C)c1 777,C1(C)(C(=O)Nc2cccc(NC(c3c(C)nn(C)c3)=O)c2)CC2(C1)CC(F)(F)C2 778,N1(C(c2c(C(C)C)sc(Cl)n2)=O)CC2(CCN(C(c3ccns3)=O)CC2)CC1C 779,C1(NC(CN(C)C(C2CCC2)=O)=O)CCC(CC(N2CCCC2CO)=O)CC1 780,CCC(F)(F)C(C)(C)C(=O)NC1CCCCCC1NC(=O)CC1CCN(C)CC1 781,Cc1cnc(CCCC(=O)NC(CNC(C2(Oc3ccccc3)CC2)=O)CO)o1 782,C1(C(=O)NCC(C)NC(C2CCC3(C2)N=N3)=O)CC2CCCC(C1)C2 783,C#CCCN=C(NCC(c1cc(C)oc1C)C)NCC(O)C1(C)CC1 784,Cc1cccc(CC(=O)NC2CC(CNC(C3CC4(CSC4)C3)=O)C2(C)C)c1 785,C1(NC(c2cn(CC)nc2)=O)CC2CN(C(C3CCS(=O)(=O)C3)=O)CC12 786,C=CCCCCC(=O)N1C2CCC1C(C(=O)N(C)CC1CCCOC1)C2 787,Cc1cc(Br)oc1C(N1CCC(Cn2cc(CC(O)C3CC3)nn2)CC1)=O 788,S(=O)(=O)(c1ccc(=NC(CCO)C2CCC2)[nH]c1)NCCCc1c(C)cccn1 789,C1(c2cn(CCN(C(CC(C)(C)SC)=O)CC)nn2)COc2ccccc2C1 790,c1(CCNC(=O)CCC2(NC(C3CCCCO3)=O)CCC2)ncccc1F 791,C1(CNC(C2CCN(C(C)=O)C2)=O)CCC(F)(CNC(=O)C(=O)NC(C)C)CC1 792,N1(C(CCCOCCC)=O)CC(O)CC1C(=O)Nc1cnccc1C1CC1 793,N1(C(C=C(C)C)=O)CCN(C(c2ccc(C(C)(C)C)cc2C)=O)C(C(F)(F)F)C1 794,CCCCC(C)CCC(=O)N(CCN(C(c1cc2nnn(C)c2s1)=O)CC)CC 795,C1(C(=O)NC2CCN(C(c3cc(C)nn3CC(F)F)=O)C2)CCC(=C(F)F)CC1 796,N1(C(C(CC)(C)CC)=O)CCCC2(C1)C(NC(=O)C(C)SC)CCN2C 797,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC1CCN(C(CSCC(=O)OC)=O)C(C)C1 798,c1(C(N2C(COC)CN(C(C3(O)CC3(C)C)=O)CC2)=O)nc(C)n2ccccc12 799,c1(C(=O)NC23CCN(C(c4ccc(Br)o4)=O)CC2C3)ccc2occc2c1 800,CCN=C(NCCOCCNC(C1CCC(NC(=O)C2CC2)C1)=O)NC(C)(C)C 801,c1(OC(C(=O)NC2C(CNC(CCC=CCC=C)=O)C2)CC)cccc(C)c1 802,c1(CC)ccccc1C(N1CCCC(CN(C(=O)COCCOC)CC)C1)=O 803,c1(C(N(C2CN(C(CSCC=C)=O)CC2F)C)=O)cc(Cl)c(F)cc1C 804,c1(C(=O)NCC(CN(C(c2c(C)nn(C)n2)=O)C)(C)C)nc2ncccn2n1 805,C1(F)(CNC(C2(OCC)CCOC2)=O)CCCN(C(=O)C=Cc2ccsc2)CC1 806,C(CC(C(C)(C)C)NC(=O)CCC1CCC1)N(C(CC(=O)N(C)C)=O)C 807,C1(NC(CSc2n(C)c(=O)n(-c3ccccc3)n2)=O)CNCCS(=O)(=O)C1 808,Cc1ncc(CC(N2CCC(N(C(=O)C=Cc3cn[nH]c3)CCO)C2)=O)[nH]1 809,Cc1cccc(C(N2CCC(C(=O)N(CC(O)C(C)(C)C)C)C23CC3)=O)c1C#N 810,CCC(CC(C)C)C(=O)N(C)CC1COCCN1C(c1nn[nH]c1Cl)=O 811,S(=O)(=O)(c1ccc(Br)cc1NCc1ncc(Cl)cn1)NC(c1ccnn1C)C 812,N1(C(C2C(CC)CCN2C(c2ccc(N)cn2)=O)=O)CCC2(CCCO2)CC1 813,N1(C(C(C(C)C)N(CC)CC)=O)CC2(CCC(CNC(=O)Cc3ccco3)O2)C1 814,N1(C(C(CC)F)=O)CC2CC(N(C)C(c3c(-c4ccccc4)cnn3C)=O)C1C2 815,N1(C(CSCCOC)=O)CCCC2C1CCN2C(c1ccc2ccn(C)c2c1)=O 816,c1(OC)cccnc1C(=O)NC1COCC1NC(c1ccc(=O)oc1)=O 817,c1(C(=O)NCC(CN(C(C2(C)CNC(=O)C2)=O)CC)(C)C)ccc(C(C)=O)cc1 818,C(=O)(C(F)(F)C(F)(F)F)NC1(C)CN(C(=O)COCc2ccccc2)C1 819,C1(NC(c2ccc(Br)o2)=O)CC2CCC(C1)N2C(=O)CC1CCC(F)(F)CO1 820,C1(OC(C2CCN(c3ccccc3Cl)C2)=O)C=CCCCCC1 821,c1(C(c2n(CCCOC)nnn2)NCc2nnnn2C)ccncc1Br 822,CCC(C)(CO)C(=O)NCC1CC2CN(C(c3oc(C4CC4)nc3C)=O)CC12 823,C1(N(C(CN(CC)CC)=O)C)CCCC2CN(C(=O)CCc3cn(C)nn3)CC12 824,c1(C(N(C2CCN(C(=O)CN(C)S(N)(=O)=O)C2)C)=O)cccc2c1OCO2 825,C(C(=O)N=c1cc(C)n(C)[nH]1)C1(C)CCN(C(c2c(C)cc(SC)o2)=O)C1 826,c1(C(=O)NCC(C)(C)NC(c2c[nH]ccc2=N)=O)cccc2c1CCOC2 827,C(CS(=O)(=O)NC1CCC(O)C1)NS(CC)(=O)=O 828,C(=O)(C(CCC(C)C)NC(c1ccncc1O)=O)N1C(COC)CCC1 829,c1(C(=O)NC2C(F)CCN(C(Cc3c(C)n(C)nc3)=O)C2)n[nH]c2c1CSCC2 830,Cc1nccc(C(=O)NCc2cc(C(=O)NC3CCCC3C)n(C)n2)n1 831,c1(C(=O)NC2C3CN(C(COCC)=O)C2CC3)cc2ccc(NC(C)C)cc2[nH]1 832,N1(C(c2c(C)nc(CO)s2)=O)CCN(C)C(CNC(C2CC(C)(C)CN2C)=O)C1 833,c1(-c2ccc(C(N(C)CC3CC(=O)CCC(=O)N3)=O)cc2)cc2ccccc2[nH]1 834,c1(C(N2CC3C(CNC(CC4(NC(C)=O)CC4)=O)(C3)C2)=O)cc(C(C)C)n(C)n1 835,C(=O)(C(F)(F)CC(C)C)N1CCCC(CC)(NC(=O)Cn2ccc([N+](=O)[O-])n2)C1 836,c1(OC)ccnc(C2CCN(C(=O)C(N3CCNC3=O)C)C2)c1 837,N1(C(c2cc(C)c(Cl)s2)=O)CC(N(C(=O)CCc2ccc(=N)[nH]c2)C)C(C)(C)C1 838,c1(CN2C(C(=O)Nc3c(C#N)ncc(C)n3)COCC2)ccc2nc(C)oc2c1 839,C1(NC(Cn2ncc(C)c2)=O)CCC(C)N(C(=O)Cc2cncn2C)C1 840,C12(CNC(C3C(CC)C3)=O)CCCC1N(C(C1CCC(=O)N(C)C1)=O)CCC2 841,c1(-c2cc(C#N)c(F)cc2)ccc2c(c1)CCN(C(=O)NCCCCl)C2 842,CC1CCC(C)(C(N2CCN(c3nccc(C#N)n3)C(CCO)C2)=O)CC1 843,N1(C(C(C)N(C(C)=O)C)=O)CC2C(CNC(c3cc[nH]c3C3CCC3)=O)C2C1 844,N1(C(C2CC(C#N)C2)=O)CCCC2(NC(=O)Cc3cc(O)nnc3O)CCCC12 845,n1(CC(=O)NC(CC)CNC(=O)C=CCF)nnc(-c2ccsc2)n1 846,Cc1[nH]cc([N+](=O)[O-])c(=O)c1C(=O)NC1CCCC1NC(=O)C1=CCOC1 847,c1(C(N2CCC(O)(CN(C(C(CC)O)=O)C)C2)=O)cnc2ccccn2c1=O 848,C#CC1CC(NC(=O)OC(C)(C)C)(NC(=O)NCCS(=O)(=O)C2CC2)C1 849,Cc1cc(F)c(C(=O)N(C2CN(C(=O)C(C)(C)c3cccs3)C2)C)cc1F 850,c1(CC(=O)NCC(CC)NC(=O)C(C(C)C)NC(=O)OCC)ccc(C)cc1Cl 851,C(=O)(C(C)C(O)CC)NCC(CN(C(c1nc(N(C)C)nc(=N)[nH]1)=O)CC)(C)C 852,c1(C(=O)NCC(C)NC(c2c(SC)cccc2)=O)cnn2c(C)ccnc12 853,C(=O)(C1CCCc2n[nH]cc21)N1CC(CNC(C(C)(C)N(C)C)=O)C(C)(C)CC1 854,c1(C(=O)OC)ccc(NC(=O)CN2CCCN(C(=O)CC(C)C)CC2)c(C#N)c1 855,c1(C(=O)NC2(CF)CCN(C(CN(C)C3CC3)=O)C2)nn(C)c(Cl)c1Cl 856,c1(C(=O)NCC(CN(C)C(C2COC(=O)N2)=O)(C)C)cccc[n+]1[O-] 857,c1(C(N2C(CNC(CC(=O)NCC)=O)CCCC2)=O)ccc(C)cc1Br 858,c1(C(=O)NCC(CCC)C(=O)NCc2scnc2C)n[nH]c2ccccc12 859,CC1CCCC(C)N1C(N1CCN(C(c2ccc(CC#N)cc2)=O)CC1)=O 860,c1(CC(N2CCN(C(CCC=C)=O)CC2CF)=O)cc(OC)c(OC)c(OC)c1 861,c1(OCC#C)ccc(C(=O)N(CC(=O)OCC)CC)cc1.c1(CN)ccccc1CO 862,c1(C(=O)NC2C(NC(=O)CCN3CCOC3=O)CC2)ccc(OC2CCC2)cn1 863,O=C(C1SCCc2sccc21)N1CC(c2cn(CC3CCOCC3)nn2)C1 864,N1(C(c2ccc(C)c(C)n2)=O)CC=C(C(=O)N2CCC(CC3CC3)C2)CC1 865,c1(C(=O)NC(CCN(C)C)C(=O)NC2CCN(CCF)C2)ccnc(O)c1F 866,c1(C(N(C2CCCCN(C(=O)CN3CC4CC4C3)C2)C)=O)nnc(O)cc1O 867,C1(CNC(C2C(C)(C)C2)=O)CCC2(CCN(C(c3n[nH]cc3[N+](=O)[O-])=O)CC2)O1 868,c1(OC)cc(C(C)NC(=O)Nc2c(OC)ccc(F)c2OC)c(F)cc1F 869,C1(C(=O)NCC2N(CC)CCC2)CC2(CCC2)CN1C(C1CN(C)CC(C)O1)=O 870,c1(N(C)C)ccc(-c2cccc(NC(C3(C(C)(F)F)CCC3)=O)n2)cc1 871,C1(NC(CC(C=C)(C)C)=O)CC2CC(C1)N(C(=O)CC(=O)N(C)C)C2 872,N1(C(c2on(C)c(=O)c2)=O)CCC(NC(=O)CCc2ccccn2)CC(C)(C)C1 873,N1(C(CCN(C(c2ccc(CC)cn2)=O)CCO)=O)CC(=O)NC2(CC2)C1 874,N1(C(c2cc(C)sc2)=O)CC(CNC(C2CCCC(C)O2)=O)CC1C 875,C(=O)(C1=Cc2cc(F)ccc2OC1)NC1C(NC(CSC(C)(C)C)=O)C1 876,c1(NC2CN(C(C(C)=C(C)C)=O)CC23CCC3)cc(C)ccc1[N+](=O)[O-] 877,C1(CNC(c2ccc(CC)o2)=O)CCCCN(C(=O)C=C(C)C2CC2)C1 878,N1(CC(N2CCOCC(NC(C(CC)O)=O)C2)=O)CCc2ccccc21 879,C1(C(=O)Nc2cc(C)c(Br)s2)CN(C(c2cc(Cl)ncc2Br)=O)CCC1(F)F 880,C(C1=CCCN(C(C2COCOC2)=O)C1)NC(Cc1c(C)nsc1)=O 881,N1(C(C(CO)N(C)C)=O)CCC(C)(CCNC(C2(CO)CCCCO2)=O)C1 882,N1(CCC(N2CCC(CNC(COCCC)=O)C(C)C2)=O)C(=O)NC(C)(C)C1=O 883,CC1(C)CCCCCC1NC(=O)C(CNC(C1OC2CCC1C2)=O)C(C)(C)C 884,C1(C(=O)NC2CCC(O)CC2)C2CC(CC2F)N1C(=O)CC1(O)CCC1 885,N#Cc1c(C(N2CC3CC2CN3C(c2ccc(I)c(O)c2)=O)=O)cccc1Cl 886,N1(C(=O)NC)CCC(C(=O)NCC2CCN2C(c2ncsc2C(F)(F)F)=O)CC1 887,N1(C(C2(CC)CCN(C(C3CC4C=CC3CC4)=O)C2)=O)CCC2(CCCCC2)C1 888,C1(CCC)(NC(=O)CC2CC(O)CN2C(c2cccnn2)=O)CCNC1=O 889,N1(C(COCC(=O)NC)=O)CC(NC(=O)CSC2CCCCO2)C(CO)C1 890,C1(CNC(C(=O)NC(C)C)=O)CC2(CCC2)CN1C(C1CCCC1C(C)C)=O 891,c1(C(N2CC(NC(CC3N(CC)CCC3)=O)C2)=O)ccc(C(C)=O)cc1C 892,c1(OCC)cc(-c2cnccc2C(=O)NCCc2ccc(F)cc2)ccc1F 893,C1(C(N(CC(F)F)C)=O)C(CNC(C2CCCS2)=O)C1(C)C 894,c1(C(N2CCC(OCCNC(C3(CC)CCOC3)=O)C2)=O)c([N+](=O)[O-])cnn1C 895,N1(C(CN(S(C)(=O)=O)C)=O)CCN(C(=O)CC2OCCC2(C)C)C2COCC12 896,S(=O)(=O)(C1CCC2(CC1)CC2)N(C)Cc1cc(Br)cn1C 897,c1(C(=O)NCCCN(C)C(c2ccc(CC3CC3)s2)=O)ccc2c(c1)N(C)CC2 898,N1(C(c2c(C)c(C3CC3)on2)=O)CC2CCCC1C2CNC(=O)Cn1cncn1 899,Cc1cc(C(=O)NC2CC3CC2N(C(=O)COCc2cc(C)on2)C3)nc(C)c1 900,c1(C(N2CCN(C(COCC(C)(C)C)=O)CC2C2CC2)=O)cc2c(s1)CCOC2 901,CC1=C(C(=O)N(CCCNC(C2CN(S(C)(=O)=O)C2)=O)C)CCO1 902,N1(C(C(C(CC)C)O)=O)CC2CCN(C(C3C4(CC4)C34CC4)=O)CC2C1 903,c1(C(N2CCC3CN(C(CCCOC)=O)CC32)=O)cc2cc(C)ccc2[nH]1 904,CCC(C)(F)C(=O)NC(C)CNC(C1(Sc2ccccc2)CC1)=O 905,O=C(CC1=CCCC1)NCc1ncccc1C(=O)NC1CCCCC12CC2 906,c1(N(CCCCN(C(=O)CC2COC(=O)C2)C)C)nnc(C2CC2)o1 907,CC1(C)CC2CC(C)(CN2C(c2cc3ccncc3[nH]2)=O)C1 908,C1(OCCC(=O)NC(CCNC(Cn2c(C)ncc2)=O)(C)C)CCN(C)CC1 909,c1(OC)cc(O)ncc1C(=O)NC1CN(C(c2n[nH]c3c2COC3)=O)CC1SC 910,CCC(CC)C(=O)N1CC(O)CC1CNC(C1CCCN(c2nccs2)C1)=O 911,C(=O)(C(CO)C(F)(F)F)NC(C(=O)NCC1C(C)(C)CC(=O)O1)COC(C)(C)C 912,c1(C(N2CC(CCNC(C(CC(C)C)C)=O)OCC2)=O)cc2ccccc2cn1 913,c1(C(=O)NC2CCCCN(C(C3OCCN(C)C3)=O)C2)cncc2ncccc12 914,C#CC1(C(=O)NCC(C)C(C)O)CCN(C(=O)COCCC(C)C)C1 915,c1(CNc2cc(NC(c3nccs3)C)ncn2)cc([N+](=O)[O-])ccc1Cl 916,CCC(CCCC(=O)N=c1ccn(C)[nH]1)NC(=O)COCCF 917,N1(C(c2cccnc2)=O)CCC2C1CCCN2C(C12CC(CO1)C2)=O 918,N1(C(=O)NCCCC2CC2(F)F)CC2CCCCC12c1ccccc1 919,C(CCC(O)C(=O)NC1CCCCCC1F)NC(CC1(N(C)C)CCC1)=O 920,C1(CNC(CCN(C(=O)Cc2cn(C)nc2C)CC)=O)CC(F)(F)CO1 921,N1(C(c2c(CC)nc(C)o2)=O)CCC(NC(c2cc(Cl)cs2)=O)C(C)(C)C1 922,CC(C)C(C)(C)C(=O)NC1CN(C(=O)CC2CCCN(C(C)C)C2)CC1O 923,CC#CCCCC(=O)NC(CCSC)C(=O)NCCNC(=O)CCC.OC 924,Cc1nc(NC(c2nnnn2C2(C)CC2)(C)COC(C)(C)C)sc1C 925,N1(C(c2c(N)c(F)cc(F)c2)=O)CCC2CN(C(c3ccnnc3)=O)CCC12 926,c1(C(N2C(CCNC(c3c(CC)scn3)=O)CSCC2)=O)cc(F)c(O)c(F)c1 927,c1(C(=O)NC2C(NC(C(COC)N(C)C)=O)CCCC2)cc(Cl)c(OC)cc1C 928,N1(C(c2c(N)cc(C)cc2F)=O)CC(NC(c2cscn2)=O)CC12CCOCC2 929,Cc1nc(C(N2CCC(C)(NC(c3cc(C(C)(C)C)c[nH]3)=O)C2)=O)c(C)o1 930,CC(C)CC(CNC(C1CCCCC(=O)C1)=O)C(=O)NCc1nn(C)cc1CO 931,c1(C(N2C(CNC(C(C)(C)c3ccno3)=O)CCC2)=O)c[nH]c2ccncc12 932,c1(C2C(C(=O)NCCN(C(=O)Cc3ccnn3C)CCC)CC2)nnc(S)n1C 933,c1(C(N2CC(F)(CNC(c3cncc(C#C)c3)=O)C2)=O)cc2cc(Cl)cnc2[nH]1 934,C(=O)(C1CCCc2n[nH]cc21)NCC1(CN(C(C(C(CC)(F)F)(C)C)=O)C)CC1 935,CC1(C)CC(c2nnnn2CC2CCOCC2)(NCC(F)C2CCC2)CS1 936,C(CCC(O)C(=O)N1CC=CC1C(=O)N(C)C)NC(CC(C)=C(C)C)=O 937,c1(N2C3CC(CN(C(c4ccc5ncnn5c4)=O)C3)C2)cccc(F)c1[N+](=O)[O-] 938,N1(C(c2ccc(C)c(O)c2)=O)C2CCC(C(=O)NCCOC(C)C)C1CC2 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1137,CCCCC(CC)C(=O)N1CCCC1C(N1CCSC2(CCC2)C1)=O 1138,Cc1cnc(C(=O)NCC(CO)NC(c2cc(F)cc(F)c2)=O)c(C)c1 1139,N1(C(C2C(C)OC(=O)N2)=O)CCC(CNC(=O)CNS(N)(=O)=O)C(O)C1 1140,C12(CNC(C(CC)CN(C)C)=O)CCC(CN(C(=O)C=Cc3ccc(C)o3)C1)C2 1141,c1(N(CC(CN(C)C(C2CCCC3CC23)=O)O)C)ccc(C#N)c(C(F)(F)F)c1 1142,C1(C)(OC(C=CC)=O)CCCC(F)(F)C1.N12CC(CC1=O)NC(=O)C(=O)N1CC2C1 1143,Cc1ccc(CCCCC(=O)NC(CNC(c2cc(C)ncn2)=O)CO)cc1 1144,C1(CNC(C(COC)C)=O)COC(C)(C)CN1C(=O)CC1(N(C)C)CC1 1145,C=CCC(C)(CNC(=O)C(CNC(C1(COC)CCCC1)=O)C(C)C)CO 1146,CC1(CNC(C2C(F)(F)C23CCC3)=O)CCN(C(C2C3CCCC23)=O)CC1 1147,C12(NC(c3c(Cl)ccc(-n4cc(CCOC)nn4)c3)=O)CCCCC1NC(=O)C2 1148,c1(CSC)cc(C(=O)NC(CCNC(=O)Cc2csc(C)n2)C(C)C)ccc1F 1149,C1(C(N(C2CC(C)C2)C)=O)CCOC1CNC(=O)CCc1cnccn1 1150,C12(CNC(COCC(=O)NC)=O)CC1CN(C(=O)CNC(=O)CC(C)(C)C)C2 1151,Cc1cc(=NC(C)c2ccc(F)c(Br)c2)[nH]c(N(C)Cc2cccn2C)n1 1152,Cc1cnc(F)c(CNC(=O)CC(C(F)F)NC(C23CSCC2C3)=O)c1 1153,Cc1cc(C(N2CC(N(C)C(C3CC3c3ccc(Cl)nc3)=O)C2)=O)nn1C(C)C 1154,c1(C(C(N2CCC(CNC(c3ccoc3)=O)C2)=O)=O)ccc(F)cc1F 1155,CC1CCC(NC(C2CC3CCC3C2)=O)CN1C(C1CCCO1)=O 1156,c1(C(N2C(CNC(c3c(C)onc3Br)=O)CCC2)=O)ccc(C)n(C)c1=O 1157,C(=O)(C(F)(F)C(F)(F)F)NCC1N(C(C2CC(C)(C)C2C(F)(F)F)=O)CCC1 1158,CCCC(C(=O)N(CC(C)NC(c1[nH]nnc1C)=O)CC)NC(C)=O 1159,Cc1nn(C)c(C)c1OCCOCCNC(=O)Nc1ccc(-c2nn[nH]n2)cc1 1160,C1(C(=O)NCc2cccc(NC(C(C)(C)F)=O)c2)CCn2cncc2C1 1161,O=C1NCCCC12CCCN(C(=NCCc1ccccn1)NCC1CCCS1)C2 1162,c1(CNC2CC(NC(c3nccnc3Cl)=O)C2)ccccc1N1CCOCC1 1163,N1(CC)CCC1C(=O)NC1CC(C(C)NC(=O)Cc2ccco2)C1 1164,c1(NC(C2(CNC(COC(CC)(C)C)=O)CC2)=O)c(SC)noc1C 1165,c1(C(N2CCCN(C(c3n(C(C)C)ccn3)=O)CC2)=O)ccc2cnoc2c1 1166,O=C(C1=COCCC1)NCC12CC1CN(C(c1ccccc1C1CC1)=O)C2 1167,C1(NC(C(C)Oc2ccc(Cl)cc2Cl)=O)CCN(C(=O)CC(F)F)C12CCC2 1168,N1(C(CSCCOC)=O)CCCN(C(C2(NC(C)=O)CCCOC2)=O)C(C)C1 1169,c1(CCCOC)cn(C(c2ccccn2)CNC(c2ccncc2)=O)nn1 1170,CC1CCOCC1C(=O)NCC1CCC(C(=O)NCCn2ccc(=O)cc2)O1 1171,C1(NC(C(C)NC(C=C)=O)=O)CC2CC1CN2C(c1cncc(Cl)c1)=O 1172,n1(CC)nc(C(=O)N(CC(C)CNC(=O)C(C)(C)c2ccsc2)C)c(C)n1 1173,C(CC(C(C)C)NC(c1ccn(C)c1C1CCC1)=O)NC(C(=C(C)C1CC1)F)=O 1174,c1(C(=O)NCC2(F)CN(C(c3cc(CC)[nH]n3)=O)C2)cccc2nc(O)n(C)c12 1175,c1(NC(c2ccc(-c3ccc(F)c(O)c3)cn2)=O)cc(Cl)cc(Cl)c1O 1176,C(=O)(C(Cn1ccnn1)NC(C)=O)NCC(C)N(C(c1cc(Cl)no1)=O)CC 1177,C1(C)(C(N(CC(CC)NC(=O)CCc2nnc(C)n2C)CC)=O)CCC(=O)N1 1178,C1(CC(=O)NCC2CN(C(c3c(C)nnn3C)=O)CC2O)CCC(C)(C)CC1 1179,c1(OC)cccc2[nH]c(C(=O)N(CCCN(C)CC(C34CSC(C3)C4)=O)C)cc12 1180,N1(C(C(c2scc(C)n2)C)=O)CCC(NC(=O)CC(C)(F)F)C12CC2 1181,C(N=c1nc2c(F)c[nH]cc-2o1)C1(C(=O)OC)CCCC1 1182,c1(C(N2C(CC)CN(C(c3[nH]c(O)nc3C)=O)CC2)=O)cccc2cncn12 1183,c1(OC)nc(C(=O)NC2CC(O)CN(C(=O)Cc3cnc[nH]3)C2)cc(O)n1 1184,CCCC(C(=O)NCCC1(O)CCN(C(c2cnc(C)[nH]2)=O)C1)OCC 1185,N1(C(C(C=C=C)C)=O)CCN(C(C2CC(S(C)(=O)=O)C2)=O)C(CCOC)C1 1186,c1(C(=O)NCC2(CNC(C(C3CC3)OC)=O)CCC2)cncc2nc(C)[nH]c12 1187,c1(OC)cccc2c(C(=O)NC3CN(C(c4cncc5sccc45)=O)C3)n[nH]c12 1188,c1(C(=O)NCC(CC=C)NC(=O)CNC=O)ccc(=O)n(C)c1 1189,CC1=C(C(=O)N2CCC(C(C)CNC(=O)C(O)(C3CC3)C3CC3)CC2)SCCO1 1190,c1(C(N2C(CNC(CC)=O)C(C)CC2)=O)cc(Br)c([N+](=O)[O-])[nH]1 1191,C(CCC(C)C(=O)NC(C)CC1CN(C(C2(C(=O)OC)CC2)=O)C1)OC 1192,Cc1nnccc1C(=O)N(CC(C)O)CCNC(=O)CC1(O)CCC1 1193,c1(CNC(c2ccc(Cl)s2)=O)ccccc1CNC(C1CC2CC1C2)=O 1194,C1(NC(C2CCN(C(CC)=O)C2)=O)CC(C(C)C)=NO1.C12(CC1)CCN2 1195,C#Cc1ccccc1CC(=O)NCCCN(C(=O)CC(C)OC)C 1196,CN1C(CNC(=O)N(CC(c2cccs2)O)C2CC2)CCS1(=O)=O 1197,S(=O)(=O)(c1cccc(Br)c1F)N1CC2CCN(C(C(C)OC)=O)C2CC1 1198,C12(NC(C(C)OCOC)=O)CC(C(N3CCC3N3CCNC3=O)=O)(C1)C2 1199,Cc1ncc(Br)c(NC2CN(C(c3ccccc3I)=O)CCC2F)n1 1200,c1(C(C)(C)C)cc(NC(=O)C(=O)NC2CCC(Cc3ccccc3)C2)cc(O)c1 1201,C(=O)(CCCC(C)(C)NC(C1CCC1C#N)=O)NC(C)CC1CC1 1202,C1(C(=O)NCC2CCCN2C(c2sc(C)cc2Cl)=O)(OCC)CCSCC1 1203,c1(C(=O)NC2CN(C3CCC3)C2)c[nH]c2cnc(Cl)cc12 1204,CC(CC(F)(F)F)C(=O)N1CCN(C(=O)COc2cccc(Cl)c2)CC1CO 1205,C1(NC(c2cc(CC)ncn2)=O)CN(C(=O)Cc2csc(Cl)c2)C2(CCOC2)C1 1206,C(C(C)(O)CC(=O)NC(CCF)C(=O)N(C)Cc1ncnn1C)OC 1207,C1(NC(CCC2CCC(NC(C3=NOC(C)C3)=O)C2)=O)CC(C)CC(C)(C)C1 1208,N1(C(c2c(C)cc(C)[nH]2)=O)CC2CC3CC2C1C3NC(=O)N.c1cn[nH]c1C(F)(F)F 1209,C(=O)(CCCCC(=O)NC)NC(C)COC.CCC1CC(=O)O1 1210,c1(CN=[N+]=[N-])ccc(C(=O)NC(CNC(c2ccncc2O)=O)C(C)(C)C)cc1 1211,C12(NC(c3nccc(Cl)c3F)=O)CCCC1CN(C(=O)CC(F)F)C2 1212,CCC(CC)CC(F)C(=O)NC1(C)CCCCC1C(=O)N(CC1CC1)CC1CC1 1213,c1(C(=O)NC(C(C)NC(C(C=CCCC)O)=O)(C)C)ccc(O)c(C(C)(C)C)c1 1214,N1(C(CCNC(C)=O)=O)CCC(C2CCCN(C(=O)C(F)=C3CCC3)C2)C1 1215,C1(F)(C(C)CNC(=O)CCC2CC2C2CCCCC2)CC(C(=O)O)C1 1216,C1(NC(C(C)SC(C)C)=O)CN(C(c2cnc3sccn23)=O)CC12CCC2 1217,c1(NC(c2sccc2NC(C2CCCO2)=O)=O)ccc(OC(F)F)cn1 1218,c1(C(N2CCC(CC)(NC(c3cnoc3)=O)C2)=O)cc2cccnc2[nH]1 1219,C(=O)(CC(C(F)(F)F)OC)NCC1N(C(C(=O)OCC)=O)CC1 1220,C1(NC(CN(C)C2CC2)=O)CC2(CCC(NC(c3c(F)ccc(F)c3O)=O)CC2)C1 1221,N(C(=NCCC(C)=O)NCc1cccc(C(F)(F)F)n1)C(CC)CO 1222,CC1CC2CN(C(C3CC3[N+](=O)[O-])=O)CC2N1C(c1ccnc(C2CC2)c1)=O 1223,c1(C(C)C)nnc2n1CC(CN1CCN(C)CC1c1ccccc1)CC2 1224,CC1CN(C(=O)CN(C(=O)C=CC(C)(C)C)C2CCC2)Cc2nncn21 1225,CCCCN=C(NCCc1cccc(SC)c1)NCCc1ccc(F)c(F)c1F 1226,C1(C(=O)NC(C2CCCCCC2)C)CCN(C(=O)c2ccc(F)cn2)O1 1227,c1(-c2c(C)c(CO)ccc2)ccc2sc(C(=O)Nc3cccnc3O)cc2c1 1228,C1(O)(CNC(C(COC)(C)OC)=O)CCN(C(=O)C(O)c2cnc[nH]2)CC1 1229,c1(OCC)ccc(CN2CC3CN(C(c4ncsc4Br)=O)CC23)cc1OCC 1230,c1(CC(=O)NC2CN(C(c3c(C)ccs3)=O)CC2C)c[nH]c2c(F)cccc12 1231,C1(N(C(c2ccc(Br)c(F)c2)CC)C=O)CC2CCC(C1)S2 1232,C1(NC(C=NOC)=O)CCCC(CNC(c2cc(Br)c(Cl)s2)=O)C1 1233,C1(C(N(CCC#C)CC)=O)(C(C)C)CCN(C(C2(CF)CC(=O)C2)=O)C1 1234,c1(C(N2C(CC(N3C(C)(CCC)CC3)=O)CCC2)=O)ccc(C#N)s1 1235,N1(C(C2CC(NC(Cc3n(C)ccc3)=O)C(O)C2)=O)CC2(C1)CC2(F)F 1236,N1(C(C(F)=C(C)C)=O)CCC2(CCCN2C(=O)CCCc2ccc(Cl)c(Cl)c2)C1 1237,c1(C(=O)NCCn2c(CC)ncc2)cc(C2CCCC2)n(C)c1C 1238,c1(C(=O)NCC2N(C(C(CCC)C#N)=O)CC=C2)[nH]c2ccccc2c1OC 1239,C(=O)(CCC(F)(F)C(=O)N(C)CCN(C)C(C12CCCCC1C2(F)F)=O)OCC 1240,C(=O)(CC(CC)C(C)C)NCc1ccc(CNC(c2cncc(C#C)c2)=O)cc1 1241,c1(C(=O)NC2C(CNC(C(C)C(F)(F)F)=O)CC2)cccc2nnn(C)c12 1242,c1(OC)ccc2c(N(C3CC(N)C3)Cc3ccc(O)cc3C)ncnc2c1 1243,C1(C(=O)NC)(COCCOCC#C)CCCNC1 1244,N1(CC(=O)NCCC2(O)CN(C(CC3C(=O)NC(=N)S3)=O)C2)CCC(=O)NC1=O 1245,c1(CC)ccnc(C(=O)NCC(CC(=O)N2CCC(O)C2)C2CCC2)c1 1246,c1(CNC(CCCN(C(c2c(C(C)C)cco2)=O)C)=O)cnc(O)nc1O 1247,C12(C(N(CC(C)SC)C)=O)CCC(CC1)N(C(c1ccnc(CO)c1)=O)C2 1248,CC(C(=O)NNC(=O)Cc1csc(=N)[nH]1)SCCNC(=O)OC(C)(C)C 1249,CN(C(=NCCC(=O)N1CCCC1)NCc1cccs1)CC1(C(F)(F)F)CCC1 1250,c1(CCC(c2nnnn2C)NCC2(OC)CC2)ccccc1F 1251,c1(CN2CC(C(=O)Nc3ccc(C)cc3Cl)SCC2)ncc(Br)cc1[N+](=O)[O-] 1252,C1(C(c2n(C)nnn2)Nc2ccc(Cl)cc2)CCC2(CC1)OCCCO2 1253,C1(CNC(C(C(=C)C)(C)C)=O)CC2(CO1)CN(C(c1ncc(C)cc1F)=O)C2 1254,Cc1cc(Br)cc(C)c1C(=O)OCC(N1CCCC(C(C)(C)O)C1)=O 1255,CCC(CC(=O)N1CCN(C(=O)COC2CCC2)C(C(C)C)C1)C(=O)OC 1256,N1(C(C(CC)CC2CCCC2)=O)CC2CCC1C(CN=c1ncc(OC)c[nH]1)C2 1257,c1(N2C(CCNC(C(C(COC)C)C)=O)CSCC2)ccc([N+](=O)[O-])cc1 1258,c1(N(C)CCN(C)C2CC2)nc(N2CCOC(C)(C)C2)nc2c1COCC2 1259,Cc1cc(C(=O)NC2(C)CNCC2(F)F)c(C)nn1 1260,C1(C(C)NC(C=CCOCCOC)=O)CCCN(C(c2[nH]cnc2C#N)=O)C1 1261,C(=O)(C1=C(C)N2CCN=C2S1)N1CCCC(O)(CNC(CSCC=C)=O)C1 1262,c1(C(=O)NC(C2CCN(C(C3CC=CC3)=O)C2)C)cc(F)c(F)cc1N 1263,c1(N(C2CN(C(C(C=C)c3ccccc3)=O)C2)C)nc(C)ncc1F 1264,c1(-c2n(C)ncn2)ccc(C(N2CC(O)CC2CNC(C2(CO)CC2)=O)=O)cc1 1265,N1(C(C=CCC)=O)CCC(C)C(CNC(c2cc(C(=O)OC)oc2C)=O)C1 1266,S(=O)(=O)(c1ccc(C(=O)NC2CC3(C2)CC3NC(=O)CC(C)C(F)(F)F)o1)NC 1267,c1(CCC)cc(C(=O)N(C2CCCC(NC(c3cnc(O)n3C)=O)C2)C)sc1C 1268,c1(CC(C)C)cc(C(N2CC(O)(C(C)NC(=O)CC3CC(O)C3)C2)=O)n[nH]1 1269,Cn1nccc1C=CC(N1CC(NC(=O)C(O)c2ccco2)C(F)C1)=O 1270,c1(C(=O)NCC2N(C(C(n3c(C)ccn3)C)=O)CCC2)cnc(Cl)c(F)c1N 1271,Cc1cc(NC(=O)CC2CC(C)N(C(C3COCCC3C)=O)C2)cc(C)c1F 1272,N1(C(C2(NC(c3cc(C)c(C)s3)=O)CC(F)C2)=O)CCN(C)C(CO)C1 1273,C=C(C)CC(C(=O)NCc1cnn(CCO)c1)NC(C1CCCN1C=O)=O 1274,N1(C(c2cc(CC)on2)=O)CC2CCN(C(C3(C#N)CC34CCC4)=O)CC12 1275,N1(C(c2c(CSC)cccn2)=O)CC2CC(NC(=O)Cn3cc[n+](C)c3)CC2C1 1276,C1(NC(c2c(C)snn2)=O)CCN(C(=O)C(C)(C)c2cscn2)CC1C 1277,Cc1ccc(C)c(C(=O)NCCCC(=O)NC2CCN(C(C)C)C2)c1 1278,C1(F)(C(=O)NC(c2c(C)ncs2)C)CCN(C(c2ccc(C#N)[nH]2)=O)C1 1279,Cc1ncc(C(N2CCC3(NC(c4cc(N)ccc4Cl)=O)CC3C2)=O)c(C)n1 1280,c1(C(c2n(CCC)nnn2)NCc2cncs2)cccc(C(F)(F)F)c1F 1281,C1(CNC(C2N(CC#C)CCC2)=O)CC(F)(F)CN1C(C1CN(C)CCO1)=O 1282,N1(C(c2c(CNC(c3c(=N)[nH]cnc3)=O)c[nH]n2)=O)CCCNC(=O)C12CC2 1283,N1(CCC)CC(C(N2CCCC2CN(C)C(C2CCC(=O)N2)=O)=O)CC1=O 1284,CC#CCC(C(=O)NCCC(O)C1CC1)NC(c1ccccc1OC)=O 1285,c1(C(=O)Nc2ccc(C#N)c(F)c2)cc2ncc(-c3cnoc3)cc2[nH]1 1286,C1(CC=C)(NC(c2sc(C3CC3)nc2C)=O)CCCN(C(=O)C(C)COC)C1 1287,N1(C(c2n(CC(C)C)ncc2)=O)CCN(C)C(CNC(=O)CC2CC2C)C1 1288,c1(C(=O)Nc2cccc(CO)c2F)ncn2cc(-c3ccco3)sc12 1289,c1(OC)ncc(C)cc1NC(=O)C(CN(C)C)NC(=O)CCCN1CCCC1 1290,Cc1c(F)ccc(C(=O)NC2CC3CC(NC(=O)C(C)C(C)C)CC23)c1C#N 1291,C(=O)(C(CC(C)C)NC(=O)CCCCC#N)OCC#C 1292,N1(C(C=C(CC)C)=O)CCN(C(=O)Cc2cc(C)[nH]n2)CC1C1CCCC1 1293,CCC(CC(=O)N1CC(C(=O)N(CCCC(C)C)C)C(CC)C1)C1CCC1 1294,c1(C(N2CCC(CN(C)C(c3ccn(CC#N)n3)=O)C2)=O)cnc(N(C)C)nc1 1295,C(=O)(CCC(F)(F)C(F)F)N1CCN(CCCNC(c2cnsc2)=O)CC1 1296,C1(C)(C(N(CCCNC(=O)CC(=O)Nc2nccs2)C)=O)CS(=O)(=O)C1 1297,Cc1ccc(C)c(OCC(N2CCN(C(=O)CCc3ccn(C)n3)C3CC23)=O)c1 1298,C1(NC(C(C)(C)OC(C)C)=O)CN(C(=O)CC2CCCC2)C2(CCOC2)C1 1299,N1(Cc2n(C)c(O)nn2)C2CCC1CN(C(c1cnc(-c3ccccc3)s1)=O)C2 1300,Cc1c(C(=O)NC2CN(C(C3CCC3(C)C)=O)CC2C)ccn1C(C)C 1301,C(CCSC)(C(=O)NC(C)(CNC(C12CCC(CC1)C2)=O)CO)OC 1302,N1(C(C(CC2CCCC2)NC(=O)CC(C2CC2)C2CC2)=O)CCC(CO)C(O)C1 1303,c1(C(N(C2CCN(C(=O)CCCNC(=O)OCC)C2)CCC)=O)cnc(O)n1C 1304,C1(C(N2C(C#C)CC2)=O)CN(C(c2occc2COC)=O)CC12CC2 1305,c1(C(=O)NC23CCC(CNC(=O)C4=CCCC4)(OC2)C3)cccc2ccsc12 1306,N1(C(CCc2scc(C)n2)=O)CCN(C(C2CCCC3CC23)=O)C2(CCC2)C1 1307,C1(CC)CN(C(=O)Cn2cc(C)cn2)CCC1NC(=O)C(C(F)(F)F)OC(C)=O 1308,N1(C(C(C)NC(=O)NC)=O)CC2(C)CN(C(C3(F)CCOC3C)=O)CC2(C)C1 1309,N1(CCC(N2C(CNC(c3[nH]cc(C(=O)OC)c3)=O)CC2)=O)CCOCC1C 1310,CC(C)C(C)C(=O)N1CCN(C2CCCC2NC(=O)CCC2CCOCC2)CC1 1311,C(=O)(CC(F)(F)C(F)(F)F)N1CCC(C)(CNC(C(C(C)C)n2cccc2)=O)C1 1312,N1(C(c2cc(C(C)C)on2)=O)CC(NC(C2CC2(Cl)Cl)=O)C2(CCOCC2)C1 1313,N1(C(Cc2cc(C)on2)=O)CC2CC(NC(=O)Cn3cc(Cl)cn3)C(C2)C1 1314,CCC(CC)C(C(=O)N1CCN(CCNC(C23CC(C)(CCO2)C3)=O)CC1)OC 1315,c1(CC(=O)NC2(CC=C)CN(C(C3(CSC)CCNC3=O)=O)C2)ccnc(F)c1 1316,C1(NC(C(CN(C)C)(C)C)=O)CC12CCN(C(c1sccc1I)=O)CC2 1317,N1(C(CC2(CC)CCC2)=O)CC(CC(=O)NCC2(CO)CC3CC3C2)CC1C 1318,C1(CNC(c2ccncn2)=O)CN(C(C2CC3(C2)CC(F)(F)C3)=O)CCC1(F)F 1319,N1(C(CCCOCCC)=O)CCC(C)(NC(C2CCCN(CCN(C)C)C2)=O)C1 1320,C=CCCC(C(=O)OC)NC(C1CN(C(c2cscn2)=O)C1)=O 1321,C1(CC(=O)NCC2C(CNC(C(CC)N(C)C)=O)C2)CCC2(CC1)CC2 1322,c1(C(N2C3(CCN)CC(C2)C3)=O)ccc(OC(F)(F)F)cc1F 1323,C(CCCCCN(C(=O)CCN1CCC1)C)NC(C(C)C1CCCO1)=O 1324,N1(C(CC2(C#N)CC2)=O)CCC2(CCC2NC(=O)CSc2ccccc2)CC1.C1(C)CC1 1325,C1(NC(c2cccc(C#C)c2C)=O)CC2CCC(C1F)N2C(C1(CF)CC1)=O 1326,Cc1ccc2c(c1)CC(NC(=O)N(C)C(c1cccs1)C)CO2 1327,C1=C(c2cc(N3CC4CCC3C4)cc(CN3CCCCC3)c2)CCNC1 1328,C(=O)(C1=CC2C=CC1C2)NCC1CN(C(C(c2c(C)n[nH]c2C)C)=O)CC1(F)F 1329,C1(c2nnnn2C)(NCC(C2CCOCC2)OCCOC)CCCC1CCCF 1330,N1(C(C=CSC)=O)CCCC(CNC(=O)C(F)(F)C2CCOCC2)CC1 1331,C1(CC(=O)NCCC(=O)NCC(=O)NC(C(=O)N(C)C)(C)C)CC2(CC2)CO1 1332,N1(C(c2n[nH]c(C)c2O)=O)CCC2C(C(=O)NC3(C)CCCC3(C)C)C2C1 1333,C1(c2n(CCS(CC=C)(=O)=O)c(N3CC=CCC3)nn2)Cc2cc(C)ccc2O1 1334,Cc1nc2c(o1)CCN(C(=O)C(CCOCCO)NC(c1ccoc1Cl)=O)C2 1335,c1(C(=O)NCC2C(NC(c3c(C#C)ccc(F)c3)=O)C2)csc2c(F)cccc12 1336,N1(C(CCC2CC(OC)C2)=O)CCN(C(c2ccc(O)cc2Cl)=O)C(C(C)C)C1 1337,c1(CCC)ncoc1C(N1CC(Cn2cc(-c3cnc(C4CC4)o3)nn2)C1)=O 1338,C1(NC(C=CCC)=O)COC2(CCN(C(=O)CC3(C#N)CC3)CC2)C1 1339,c1(NC(C2C3CC2N(C(=O)C(Cl)(Cl)Cl)C3)=O)cnc(Br)nc1 1340,c1(SCC)ccccc1C(N1CCC(NC(c2oc(CN(C)C)nc2C)=O)C1)=O 1341,C(CC)(C(=O)N(C)CC1CCN(C(C2(C3CCCO3)CCCC2)=O)C1)=CC 1342,C1(C(=O)NC2C=CC(C(=O)Nc3c(OC)ncnc3)C2)CCCCC(=O)N1 1343,C(=O)(C#CC1CCOCC1)NC(C1CCN(C(c2cc(Cl)cc(C)c2O)=O)C1)C 1344,C1(C(=O)NCC(C)N(C)C)CCN(C(C2(N3CCCC3)CC2)=O)C1 1345,c1(C(N2CC(CN(C(CC(C)SC)=O)C)C3(C2)CC3)=O)cc2cc(C)ccc2[nH]1 1346,c1(C(=O)NC2(C)CC(NC(c3cn(C)c(=O)cc3)=O)C2)coc2ccc(F)cc12 1347,c1(C(=O)NC(CC)(C)CNC(=O)COCc2nc(CC)no2)cc(Cl)ccc1N 1348,C(=O)(C(CS(C)(=O)=O)c1ccccc1)OCC(C(C)C)(C)C.c12ccccc1N2 1349,c1(NC(c2c(C(C)NC(CC3C(C)OCC3)=O)noc2)=O)ccc(O)cc1Cl 1350,C1(C(=O)NCC(C)CN(C)C(C2CC3CC3C2)=O)CCc2ccnn2C1 1351,C1(OC)CC(NC(c2ccsc2)=O)CN(C(c2cncc(OC(C)C)c2)=O)C1 1352,C1(C(N)=O)CN(C(C2(F)CN(C(C3(c4cccs4)CC3)=O)C2)=O)CCC1O 1353,O=C(N=c1nc(SC2CC2)s[nH]1)N1CCOC(CC2CCC2)C1 1354,CCCC(C(=O)NCC1CC2CN(C(c3ccc(Cl)cc3OC)=O)CC12)C(C)C 1355,CC#CCCCC(=O)NCc1ccc(C(=O)NC(C)CN(C)C)cc1 1356,C1(NC(C(CC)CC)=O)CC(F)(F)CC1NC(c1cc(Cl)c(Cl)s1)=O 1357,c1(C(c2ncc[nH]2)NCC(CO)NC(C(C)N(S(C)(=O)=O)CCO)=O)ccccc1 1358,C1(O)(C(N)=O)CCCN(C(C2CSCCN2C(c2cc(Cl)cs2)=O)=O)C1 1359,c1(CC(N2C(CNC(CC=CCC)=O)CC2)=O)cc2ccccc2nc1O 1360,N1(C(c2c(COC)cc[nH]2)=O)CC(NC(=O)C=C(C)C(C)(C)C)C(C)C1 1361,C1(C(=O)OC)C2C=CC(CC2)C1C(N1CCC(NCC2CC2c2cnc[nH]2)C1)=O 1362,C1(N(C(C(C=C=C)C)=O)C)CN(C(=O)C(F)(F)Cc2ccccc2)CC12CC2 1363,C1(NC(C(C)OCCCC)=O)CCC(O)CN(C(C2(c3ccn(C)n3)CC2)=O)C1 1364,c1(CNC(C(=O)Nc2c(C(=O)OC)scc2)=O)cccc(NC(C)=O)c1 1365,C1(C(N(C2(CO)CC2)C)=O)CN(C(=O)CC2CCSC2)CCC1(C)C 1366,N1(C(C(CC)C#N)=O)CC2C3CCC(C2C1)N(C(C1CC1(C)C(F)F)=O)C3 1367,CCC(C(=O)N1CCN(C)CC1C(=O)NCC1(OC)CCOC1)C(C)(C)CC 1368,C1(C(C)C)CCC(C(=O)N(C)CC2CCCN(C(C3(CO)CCCO3)=O)C2)CC1 1369,N1(CC(N2CC(CN(C)C(C3COCCO3)=O)C2)=O)CCCCC1=O 1370,c1(C(N2C(CNC(CCC#C)=O)CC(O)C2)=O)cc(OC)cc(F)c1 1371,CO[Si](C)(CCCOC(C1(CC(C)C)CC1)=O)OC 1372,C12(NC(COC(CC)C)=O)CCC(CNC(c3cn(C)c(C)n3)=O)(CC1)OC2 1373,CCCCC(C(=O)N1CCC(C)C1CNC(=O)C(C1CCOC1)OC)C(C)C 1374,N1(C(CCCOC)=O)CCCC2(NC(=O)CN(c3ccccc3)C)CC12 1375,N1(C(CCCC=C)=O)CCN(C(C23CC=CC(C2)OC3)=O)C(CC)C1 1376,c1(C(N2CC(NC(CSC(C)C)=O)C(C)(C)C2)=O)c(F)cccc1[N+](=O)[O-] 1377,c1(C(=O)NC2CC3(C2)CC(NC(C2CC2(F)Cl)=O)C3)cc2cccnn2n1 1378,CCC#CCN=c1nc(N2CCC(c3cccc(F)c3)CC2)c2c([nH]1)CCC2 1379,c1(C(=O)NCC(CO)NC(CCNC(N)=O)=O)coc2c1C(=O)NCC2 1380,c1(NCC2CC(NC(c3nc(NC(C(C)C)=O)sc3)=O)C2)ccccc1[N+](=O)[O-] 1381,CCC(CC(=O)NC(CC(F)F)C(=O)N1CCCC(C(C)C)CC1)CC(C)C 1382,CN1CC=C(CC(=O)NC2CCN(C(C3CC3C(=O)NCCO)=O)C23CCC3)CC1 1383,Cc1ccc2cc(C(N3CCCCC3CNC(C3CSCCS3)=O)=O)cnc2c1 1384,C1(C(=O)NC(C)(CNC(c2cc(C(F)(F)F)n[nH]2)=O)CO)COC2(CCC2)CO1 1385,c1(C(=O)NCC(CC)(CC)NC(CNC(CC)=O)=O)c[nH]c2c(F)cccc12 1386,C(C(O)CCNC(C1CN(C2CCOC2)C1)=O)NC(c1cccs1)=O 1387,C(=O)(C(CNC(c1ccc(C)nc1)=O)C(C)(C)C)NCCC(COC)O 1388,c1(CC(=O)NCC2(C(=O)NCC(F)CO)CCC2)cnoc1 1389,C(=O)(N=c1c(Br)c[nH]cc1Br)C1NCCN(Cc2c(O)cc(OC)c(Br)c2)C1 1390,N1(C(C(C)N(C(C=CC(=O)OCC)=O)CC)=O)CCCC(C2(C)CC2)C1 1391,N1(CCC(N2CC(OC)(CNC(c3ocnc3C)=O)C2)=O)CCCC(C(N)=O)C1 1392,C(=O)(N=c1ccn(CC(c2ccccn2)N(C)C)[nH]1)N(CC(C)(C)O)C 1393,c1(C2(C(N(CCOCCN(C(CSCC=C)=O)C)C)=O)CC2)ccccc1 1394,C(=O)(CS(=O)(=O)C(C)C)N1CC(CNC(C2CCCN(C(C)=O)C2)=O)N(C)CC1 1395,Cc1ccc(N)cc1C(N1CC2(C1)CN(C(=O)C(c1ccccc1Cl)O)C2)=O 1396,C1(C(N2C(CCNC(C(C)C3CCCC3)=O)CCCC2)=O)CCC([N+](=O)[O-])CC1 1397,C1(NC(C(c2cscn2)N(C)C)=O)CCN(C(c2cnn(C)c2)=O)C1C(C)(C)C 1398,c1(-c2cn(C(CNC(c3cc(OC)n[nH]3)=O)C)nn2)cccc(F)c1N 1399,N1(C(C2CCC(C)CC2)=O)CCOC2(CCN(C(=O)C=C3CCC3)C2)C1 1400,N1(C(c2n[nH]cc2Br)=O)CCC(C2CC2)C1CNC(C1(CCF)CCC1)=O 1401,c1(C(N(C2CCN(C(CCC(=C)C)=O)CC2)C)=O)c(Cl)cccc1[N+](=O)[O-] 1402,C(=O)(C(C)(c1ccccc1)OC(C)C)NCC(C)NC(C=CCC)=O 1403,C12(C(=O)NC(C(=O)OC)C)COCC1CN(Cc1ccc(OCCN(C)C)nc1)C2 1404,C1(C(=O)NCC2(SC)CC2)CCCN1C(C)C.C1=CC(=O)NC1(C)C 1405,C(CC(C)(C)C)(C(=O)NCCCC1(O)CCC1)NC(C(CCC)C)=O 1406,c1(SC)ccc(C(N2CC3CC3(CNC(=O)CC(C)C)C2)=O)cc1Br 1407,c1(C(=O)NC2(CC(=O)NC3CC(CC)(CC)C3)CC2)cccc(F)c1O.O 1408,N1(C(CC2ON=C(C)C2)=O)CCCC(CCNC(=O)C(c2ccc(Cl)cc2)O)C1 1409,c1(C(=O)NC2C=CC(CNC(c3n(CC)ncc3)=O)C2)c(F)cccc1F 1410,C(c1cc(F)c(F)c(F)c1)=CC(N1CCC(N(C(C(C)OC)=O)C)C1)=O 1411,N1(C(c2c(C)csn2)=O)CC(C(=O)N(C2CCCC2C#N)C)CC(C)C1 1412,C1(NC(CCn2c(C)csc2=O)=O)CC2(C1)CC(NC(C1(C3CC3)CC1)=O)C2 1413,N1(C(Cc2nc(C)on2)=O)CCC(C(N2CCOC(C(C)C)C2)=O)C2OCCC12 1414,c1(C(=O)NCCN2CCN(C(CC(C)N(C)C)=O)CC2)ccc(C#N)cc1F 1415,C(=O)(C1CCCc2n[nH]cc21)N(CC(C)NC(c1ccc(CC)cc1N)=O)C 1416,c1(C(=O)NCC(CNC(c2c(CC)nns2)=O)(C)F)ccc2ncncc2c1 1417,CON=C(C(=O)NCC1(C)CCN(C(=O)C2CC2)CC1)c1ccco1 1418,n1(C(C)(C)C)nc2c(c1C(=O)NCCCNC(c1cc(Cl)ccn1)=O)CCCC2 1419,Cn1c(=O)[nH]c(NCC2CCN(c3ccccc3Cl)C2)c(C#N)c1=O 1420,C1(CC=C)(C(=O)O)CCN(C(C2CCC(N)CC2)=O)CC1 1421,c1(C(N2CCC(C)(CNC(C3CC3F)=O)C2)=O)ccn2nnnc2c1 1422,Cc1nc(C(=O)NCC2CC2CNC(c2ccc(Br)s2)=O)cn1C 1423,c1(OCC=C)ccc(Br)cc1C(=O)NC1COCCC1O 1424,C1(C(N(C(CCNC(CNC(=O)NC)=O)C)C)=O)CC(C)CO1 1425,CC(C)(C)CC(=O)NC1CC2C(NC(=O)COC3CCCOC3)C2C1 1426,Cc1ccc(CC(=O)NCCC2(OC)CN(C(C3CCC(C(N)=O)O3)=O)C2)cc1 1427,c1(C(N(CC(N2CC(OC(N)=O)C2)=O)C2CCC2)=O)coc(CO)c1 1428,c1(C(=O)NC2CN(C(C(c3ccccc3Cl)OC)=O)C2)nsc2c(Cl)cccc12 1429,n1(CCCC)nnnc1C(CCC1CC=CCC1)NCC=C(C)C 1430,CC1CCN(C(c2cnn(-c3ccc(F)cc3)n2)=O)CC1NC(c1cnns1)=O 1431,C(=O)(CC(O)C(C)C)NCCC1(OC)CN(C(CNC(=O)OC)=O)C1 1432,C1(NC(C(CCSC)NC(CC)=O)=O)CC2CCCCCC12 1433,c1(COC)cccc(NC(C2(O)CCN(C(=O)Cc3cnn(C(C)C)c3)C2)=O)c1 1434,C(N=c1cc(C)nc(Cl)[nH]1)C1CN(C(C2(COC)CCCCO2)=O)C(C)C1 1435,C=CC(C)(O)C(=O)NCC(C)(C(C)C)NC(c1cc(Cl)sc1Cl)=O 1436,C1(C(N2CCC(C(C)NC(C3(CCN(C)C)CC3)=O)C2)=O)CCCCC(C)(C)C1 1437,CC1CCC(CC(N2CC(CC(F)C(=O)N3CCC(CCCO)C3)C2)=O)C1 1438,N1(C(c2c(C)nsc2)=O)CC(N(C)C(c2cncs2)=O)C(F)C1 1439,CCC(CC)C(C(=O)NCCC(=O)NC(CO)C(C)C)OC 1440,C=CCC(CC(C)C)C(=O)N1CCCC(C)(C)C1C(=O)NC1(CCOC)CC1 1441,CCC(c1cccc(Cl)c1)=CC(=O)NCC1CCC1NC(=O)CC1CC1 1442,CC1CCCC1(C)NC(=O)CCOCCCNC(C1CCC(N(C)C)C1)=O 1443,CC1CCCC(C(N2CCN(CCNC(=O)COCCF)CC2)=O)CC1 1444,Cc1nc(C(C)C)sc1C(=O)NC1CCC(CNC(c2n[nH]cc2F)=O)C1 1445,c1(NC(=O)Nc2cnc(C3CCOCC3)nc2)ncc(Br)c2cccnc12 1446,N1(C(C23CCC(C)(CC2)OC3)=O)CCCC2CN(C(C3CC3C3CC3)=O)CCC12 1447,C(=O)(NNc1c(Cl)cccc1Br)C1(C2C(=O)CCC2)CCC1 1448,c1(Oc2cc(C(=O)OCC)sc2C)c(Cl)ccnc1Br 1449,c1(C(=O)NC2C(C(N3C(CC)C(O)CC3)=O)CCCC2)ccc(C)c(C#N)c1 1450,C1(C#CC(=O)N2CCC(O)C2C(=O)NC2(COC(C)=O)CC2)(CC)COC1 1451,N1(C(CCC(C)(C)F)=O)CCC2(CCCN(C(=O)CC(C)(C)C3CC3)C2)C1 1452,n1(CC)cc(NC(C2CC(C)CN2Cc2cnc(N(C)C)nc2)=O)c(C)n1 1453,N1(C(=O)NC(C)(CO)C(F)F)CCC2(C1)CN(C(c1ccccc1)=O)CCO2 1454,C#CCC(C)(C(=O)NC(c1nc[nH]n1)CC)NC(=O)CC1CCC(=O)N1 1455,c1(C(N(C2CC(NC(C3CC3c3ccco3)=O)C2)C)=O)cc(Br)cnc1N 1456,c1(C(N2CC(CNC(c3cc(C)n(C)n3)=O)C(C)C2)=O)ccn2cnnc2c1 1457,c1(OC)ccc(C(=O)NCC2CC(F)(CNC(C3(F)CC3C)=O)C2)c(F)c1 1458,c1(C(=O)NCC2(F)CCC(NC(c3c(C)noc3)=O)C2)cnc2ccccn12 1459,n1(CC(N2CCCC(N(C(C(CCC)C)=O)C)C2)=O)ncc(C#N)c1Br 1460,C1(C(N(CCC(=O)NCC2(C3CC3)CCC2)CC#C)=O)CCCC(C#N)C1 1461,c1(C(N(CC(C)O)CCNC(=O)CCc2cn[nH]c2)=O)ccc(SC(F)(F)F)o1 1462,C1(C(=O)Nc2cccc(CNC(CCC)=O)c2)Cc2cc(C)c(C)cc2O1 1463,CCCCCC(O)CC(=O)NC(CNC(=O)CCOc1cccnc1)CCC 1464,C(=O)(CC1=NNC(=O)C1)NCCC(CCNC(C(C)C1CC1)=O)C 1465,N1(C(c2c(C(C)C)c[nH]n2)=O)CCC2CN(C(c3csc(C(N)=O)n3)=O)CC2C1 1466,C(=O)(C1=C(C#N)CCC1)N1CCC(OC)(CNC(C2CN(C)C2)=O)CC1 1467,C(C(=O)NCC1C2CN(C(=O)CC(C)CN(C)C)CC12)(C(C)C)n1cc(C)nc1 1468,N1(C(c2c[nH]c(=NC)s2)=O)CCN2CCN(C(=O)C(C)C3CC3)CC2C1 1469,C12(CNC(CC3CCN(C(C)=O)C3)=O)CC(NC(C3CCCSC3)=O)(CCO1)C2 1470,C1(C(=O)N(CC(O)CO)C)(CC)CCN(C(c2ccnn2COC)=O)C1 1471,C1(C(N(C(COCc2cn(CCCC)nn2)C)C)=O)CCC(OC)CC1 1472,C(=O)(C1=CS(=O)CCC1)N1CCC(C(C)NC(C(C)c2cccs2)=O)CC1 1473,Cc1cc(CN(c2cc(Cl)nc(Cl)c2)C)cc(Cl)c1 1474,O=C(C=CCN1CCCCC1)NOCC(=O)NC1CC1.C1(CC2CC2)CC1 1475,n1(CC)c(C)cc2c1CCCC2NC(=O)C(=O)NCC1OC(=O)CC1(C)C 1476,c1(OC)cc2[nH]ncc2cc1NC(=O)NC1CN2CCC1C2 1477,N1(C(C(Cn2cc(-c3nc(C4CC4)cs3)nn2)CO)COC)CCCCCC1C 1478,N1(C(C2C(COC)CC2)=O)CCc2ccccc2C1CO 1479,c1(C(=O)NC2C(CNC(CN(C(C)C)C)=O)C2)coc(Cl)n1 1480,C1(CNC(=O)C(O)C(F)F)COCCN(C(c2c[nH]nc2-c2ccccc2)=O)C1 1481,C1(CNC(=O)CCF)CC2(C1)CC(N=c1[nH]c3ccccc3o1)CCS2(=O)=O 1482,C1(NC(Cc2ccc(C)cc2)=O)CCN(C(c2ccc(C)n2C)=O)CC1C(N)=O 1483,c1(C(=O)NC(CN(C(c2cc(CC)on2)=O)C)(C)C)sc2nccnc2c1N 1484,O(NC(=O)C(F)C(C)CNC(C1(C)CC(=O)C1)=O)CCC=C 1485,CC1CCN(C(=O)C(O)CC2CCCC2)CC1CNC(c1ccc(C2CC2)nc1)=O 1486,c1(OC)cc(CN2CCC(NC(c3cccc(F)c3I)=O)C(F)C2)ccc1C 1487,CN1C(=O)CN(CC(=O)NC2CN(C(c3cnccn3)=O)CCC2C)C1=O 1488,C1(C2CCN(C(=O)C(F)=C(C)C)CC2)(NC(C=C(C)C(C)(C)C)=O)CC1 1489,N1(C(=O)C=CC2CC2)CC2(CCCC2NC(=O)C(F)(F)Cl)C1 1490,Cc1nccc(Cl)c1C(N1CC(N(C(=O)C(Cl)=CCl)C)C(C)(C)C1)=O 1491,N1(CC(=O)NCC2CC(F)(F)CN2C(=O)CCc2ccco2)CCCNS1(=O)=O 1492,c1(NC(C2N(S(c3cn(CC)nc3)(=O)=O)C3C(C2)C3)=O)ccc2oncc2c1 1493,Cc1csc(C(=O)NC2(C(=O)N(C)CC3(O)CCOC3)CC(O)C2)c1 1494,N1(C(C2CCN(C(=O)OCC)CC2)=O)CCCC(NC(C2CC(C)(O)C2)=O)C1C 1495,C1(CNC(c2c(C)n(C)cn2)=O)CC2CN(C(=O)C=Cc3ccc(Cl)cc3)CC12 1496,c1(OCCC)cccc(C(N2CC(O)CC2CNC(C2(C)CCNC2=O)=O)=O)c1 1497,C(C(C)C(F)C(=O)NCCC1NC(=O)NC1=O)NC(c1c(C)nco1)=O 1498,C1(CNC(=O)CCCN2CCCC2)CCN(C(=O)CCCC2CCC2)C12CCC2 1499,Cc1cc(C)n(CC(=O)NC2(c3cn(-n4ccccc4=O)nn3)CC(F)(F)C2)n1 1500,C1(CNC(CCNC(=O)NC)=O)(NC(=O)C(CO)NC(N)=O)CCOC1.C(C)C 1501,C1(C(=O)NCCCN(C(=O)C=C2CCN(C)CC2)CC)CCCC1(C)N(C)C 1502,C#CC1(OC(C2CCCC(OCC)C2)=O)CCC(C)(C)C1 1503,N1(C(C)C)CCC(CNC(=O)C(O)CNC(=O)C(F)=CC2CC2)C1 1504,C1(NC(Cc2cn(C)nc2)=O)CC2(C1)CN(C(C1CNC(=O)C1)=O)C2 1505,CCCCN=C(NCCN1CCCCC1=O)NC1Cc2ccccc21 1506,Cc1ccc(C=CC(=O)N(C2CCN(C(=O)C=C3CCC(C)C3)CC2)C)cn1 1507,c1(C(c2n(C(C(=O)OC)C)nnn2)NC2C(C)C2(C)C)ccc(OC)nc1 1508,C1(NC(C(C2CCCCC2)OC)=O)C2CCCN(C(=O)COC(F)F)C2C1(C)C 1509,c1(C(N(C2CCCN(C(C3CCCCN3C)=O)C2)CC)=O)[nH]c(O)nc1C 1510,c1(C(=O)NCC(c2ccccc2)N(C(C(C)OC)=O)C)ccc(O)c(Br)c1 1511,N1(C(C(CC)C(C)O)=O)CCC2CC(NC(c3cc(F)ccc3Cl)=O)CCC2C1 1512,N1(C(CC(=O)NCC#C)=O)CC2CC(NC(=O)CC3COCC3(C)C)C(C2)C1 1513,c1(C(N2CCN(C(c3c(CC)cncc3)=O)C(C)C2)=O)cc(F)cc(Cl)c1O 1514,C(=O)(C(C)CC(=C)C)NCCCCN(CCCNC(CC=C=C)=O)C 1515,C1(OCC)CN(C(=O)CC2CCC2OC)CC1CNC(=O)C=Cc1csnc1C 1516,c1(C(=O)NC(CC)CNC(=O)C(=O)NC(C)C)sc(C(C)C)nc1C 1517,CCCC(C)CCN=c1[nH]ccc(=NCCc2cc(F)ccc2C)[nH]1 1518,CC(C(=O)NC1CCCCC1CNC(=O)C(=O)NCC(F)(F)F)C(C)(F)F 1519,c1(CNC(c2cc(C)ncn2)c2n(CCCSC)nnn2)ccc2nsnc2c1 1520,Cc1[nH]c(C)c(C(=O)NC(C)CNC(c2ccoc2C2CCN(C)CC2)=O)c1C 1521,S(=O)(=O)(c1cccc(=NC2CCC(F)(F)C2)[nH]1)NCc1c(C)nc(C)c(C)n1 1522,C1(N(C)C)CC(N=c2[nH]c(N3CCc4nc(N(C)C)sc4C3)nc(=N)[nH]2)C1 1523,C(=O)(C(C(C)NC(=O)CCc1cnco1)C(C)C)NCCC(=O)OC(C)C 1524,N1(C(CC2(C)OCCO2)=O)CCN(C(C2CCC(=O)NC2)=O)CC1c1cn[nH]c1 1525,CN1C(=O)NCC1C(=O)NC1CCN(C(=O)CCSc2ccc(F)cc2)C1 1526,C1(C)(CCC(=O)Nc2c(CC)csc2)CCCN1C(=O)C(C(C)C)OCC(C)C 1527,N1(C(c2cc(C)c(Cl)cc2Cl)=O)CCC2(CC(NC(=O)CC3CC3)CO2)C1 1528,C(=O)(C#CC1CCOCC1)N1CC(NC(Cc2nnc(C)o2)=O)C2C1CCC2 1529,N1(C(C2C(=C)C2)=O)CCc2ccccc2C1CNC(c1cnn(C2CC2)c1Cl)=O 1530,C1(CN(C)C(C2CC23CC(NC(C24CCC(C2)C4)=O)C3)=O)CCCCC1(C)C 1531,C#CCC(C)(CC)C(=O)N1CCC1CNC(C1(O)CCSCC1)=O 1532,Cc1ccc2c(N(CC(F)F)C)nc(N(C)CC3CCCS3(=O)=O)nc2c1 1533,C(C)(C(CC(=O)NCCc1ccc(F)nc1)NC(=O)CCN1CCCCC1)OC 1534,C1(NC(CCc2cncc(C)c2)=O)CCN(C(=O)C(C)n2cccc2)C(C)C1 1535,CC(C(C(=O)NCC1CC1)N1CCC(C)(CNC(=O)OC(C)(C)C)CC1)C(C)(C)C 1536,C1(CNC(CC=CC=C)=O)CCCCN(C(=O)COCc2ccccn2)C1 1537,c1(CCC(=O)NC(CCNC(C2C(C(=O)OC)CCC2)=O)C)ccccc1OC 1538,CCCCCC(=O)NC(c1ccccc1)C(C)NC(c1cccnc1S)=O 1539,Cc1cc(F)ccc1CC(=O)NCC1CC(NC(=O)C(C)(C)c2ccccn2)C1 1540,N1(C(c2ncn(CC)c2)=O)CCC(NC(=O)C(N)=O)C(C)C1 1541,N1(C(CN(C)C(N)=O)=O)CCCC(O)(CCNC(=O)C(O)Cc2ccccc2)C1 1542,C1(O)(CNC(C2CCCS2)=O)CCCN(C(=O)CN2CCCC2)CC1 1543,C(=O)(C(CO)c1ccccc1)NC(C1CCN(C(=O)CCc2cc[nH]n2)C1)(C)C 1544,n1(CC)ccc(CN(C(=O)COCCNC(=O)C(C)C2CCOC2)C)n1 1545,c1(C(=O)NCCCN(C(CC2CC(CC)C2)=O)CC)ccc(F)cc1C(F)(F)F 1546,N1(C(CC(C=C)CC)=O)CCC(C(=O)N(C)Cc2ccc(C)nc2)C(C)(C)C1 1547,C1(NC(C2C=CCN(C(c3ccccc3)=O)C2)=O)CC2(CCC2)C1O 1548,C1(C(N2CCN(C(CC(n3ccc(C)n3)C)=O)CC2C)=O)CC2CCCCN2C1 1549,C1(CC(=O)NC(CNC(C(C(C)C)OC)=O)(C)C)CCC(=O)NC1=O 1550,Cc1nc2ncc(C(=O)NC(CNC(=O)Cn3cncn3)CC(C)C)cc2o1 1551,C1(NC(C23CCC(C2)C3)=O)CCCC(NC(C2(Br)CC2)=O)C1 1552,C1(CC(=O)NCC2CCC(C)C2)CCN(C(=O)C2=NNC(=O)C2)C1(C)C 1553,C#Cc1ccc(C(=O)NCC(O)CCNC(c2c[nH]cc2C)=O)cc1 1554,C(C(N=c1cc[nH]c(-c2ccc(C(C)(C)C)cc2)n1)c1cnn(C)c1)OC(C)C 1555,C1(NC(C(CCF)NC(COCCC)=O)=O)C2CCC(C2)C1C 1556,C(=O)(C#CC1CCCOC1)NC1C(C)(C)N(c2nc(C#N)ncc2Cl)CC1 1557,N1(C(C2=CCCN(C(CCC(C)=O)=O)C2)=O)CC(=O)N2CCCC2C1 1558,c1(C(C)C)cccc2c(OCC(=O)OCC3CCCO3)ccnc12.O 1559,CC(CCC(=O)N1CCC(C)(CNC(=O)COCC(C)(C)C)C1)N(C)C 1560,C1(N(C(=O)CCc2ccccc2)CC)CCCN(C(C2(Cl)CC2(F)F)=O)C1 1561,c1(CC)nn(C)c(CC(N2CCCC(NC(c3cncn3C)=O)C2C)=O)c1Br 1562,N1(C(CCCSC)=O)CC(NC(=O)C=CC2CCCCCC2)CC(C)(C)C1 1563,c1(N2CCCC(CNC(c3c(CC)c[nH]c3)=O)C2)ncnc2ccc(C)cc12 1564,c1(OC)nc(C)sc1C(=O)NCC1CCC(NC(c2ccc(C(C)C)nc2)=O)C1 1565,C1(CC(C)NC(C(C)(C)SC)=O)CC2CCC(C1)N2C(=O)CCn1ccc(=N)[nH]1 1566,C(=O)(CCCS(C)(=O)=O)N1CC(NC(C(C=C)(C)C)=O)C2C(C1)C2 1567,C1(C(=O)OCC)CC2CCC1N(C(=O)C(=O)NCc1cccc3c[nH]nc13)C2 1568,C1(CC(=O)N(C)Cc2nccs2)CCCN(C(C2CC3C=CC2C3)=O)CC1 1569,N(C(=NCCC(C)(C)C=C)N1CCN2C(CCS2(=O)=O)C1)C(C=C)C 1570,S(=O)(=O)(c1cc(C(F)(F)F)ccc1N(CCC#N)C)NCC(C)C(C)(F)F 1571,C12(CCN(C(=O)CSCCN(C)C)C1)C(=O)N2.C1(CC)CC(CN(C)C)C1 1572,CCCC(CCCNC(C1(O)CCC1)=O)NC(c1cc(CO)n(C)n1)=O 1573,c1(CCC(N2CCC(C(C)NC(=O)CCc3cnn(C)c3)C2)=O)ncc(F)cn1 1574,CC1(C)CC(NC(C2CC2F)=O)CCN(C(=O)CCc2cc(Cl)cs2)C1 1575,C12(CCOCC1)C(=O)N2.c1(C(=O)NC2CCN(CC)C2)cn(CCOC)nc1C 1576,N1(C(C(C)(F)F)=O)CCCC(C2CCN(C(C3(C#N)CC4CCC3CC4)=O)C2)C1 1577,CN=c1[nH]c(C(N2CCN(CC(C)(C)NC(C3CC34CC(O)C4)=O)CC2)=O)cs1 1578,C1(CNC(c2n(C(CC)C)ncc2)=O)CN(C(C2CC2(F)F)=O)CCC1(C)C 1579,c1(Nc2ccc(CC(C)C)cc2)nccc(=NC2CCC3C4CCC(C4)C23)[nH]1 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1668,C1(O)(CNC(c2c(C)nn(C(C)C)c2)=O)CCN(C(C2CC2F)=O)CC1 1669,C1(CC(=O)N(CC(O)CNC(c2conc2C(C)(C)C)=O)C)CCN(C)C1=O 1670,c1(CC)cc(=NC(=O)C2CCCC2NC(C2CNC(=O)CC2C)=O)[nH]n1C 1671,C(=O)(C1COc2ccccc21)N1CC2C(NC(=O)C(F)=CCCF)(CC2)C1 1672,C1(C(=O)CNC(CCN(C(=O)CC(C)n2cccn2)CC)=O)(C2CC2)CCCO1 1673,N1(C(c2cn(CC=C)nn2)=O)CCOC(CN(C(=O)CC=CC)C)C1 1674,N1(C(C2C(NC(C(C)(C)NC(C)=O)=O)C2)=O)CCN(S(C)(=O)=O)CC1 1675,CC1(C)C2CN(C(=O)CC3C4CCC(C4)N3C(=O)CC3CCC(=O)NC3)CC12 1676,C(=O)(CC(C)C(=O)OC)NCCN(C(c1ccn(C2CCOCC2)n1)=O)CC 1677,C(=O)(CC(CN(C)C)C(F)(F)F)NCCCN(C(CC1(CC=C)CCCC1)=O)C 1678,C1(C(=O)NC(C2(O)CCN(C(C3CC(O)C3)=O)C2)C)CCc2nnnn2CC1 1679,C#CCCCCCC(=O)N1CC2(CC(CC(=O)N(C(C)C3=CCCOC3)C)C2)C1 1680,c1(C(=O)NCc2ccc(C(N3CCC(CN(C)CC)C3)=O)s2)n[nH]c(C)c1Cl 1681,c1(C(N2CCC(N(C(CCC=CC)=O)CCO)C2)=O)cc(F)cc(Br)c1F 1682,c1(NC(=O)C2CC2)cncc(C(=O)NC2CCN(Cc3ccc(OC)nc3)C2)c1 1683,N1(C(C(CCC2CCC2)NC(C(=O)C2CCCC2)=O)=O)CC2(CCC(O)CC2)C1 1684,C(=O)(C(C)S(=O)(=O)C(C)C)N(CCN(C(c1c(N)sc(C)c1C)=O)C)C(C)C 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1702,N1(C(CC)=O)CCC(C)C(NC(=O)N(C(C2CCCCCCC2)C)CC)C1 1703,N1(C(c2cc(C)ns2)=O)CCC(NC(=O)Cc2ccsn2)C1C 1704,Cc1nc(O)ccc1C(N1CCC(C(C)NC(=O)C2=CCCS2)C1)=O 1705,c1(OCC(=O)NC2(CO)CN(C(CC(=O)N(C)C)=O)C2)ccc(Br)nc1 1706,c1(C(=O)Nc2c(SCC)cc(C)cc2)ccc2[nH]cc(C#N)c2c1 1707,CCC(C)C(C(=O)N1CCOCC(CNC(c2ccsc2OC)=O)C1)OC 1708,CN1CC=C(CC(=O)NCC2C=CCN2C(=O)Cc2c(O)ncnc2O)CC1 1709,C1(C)(C(=O)NC(C)CNC(=O)C(Cc2ccccc2)n2cnnn2)COCCO1 1710,c1(C(N2CCC(CCOC)(NC(CSCC=C)=O)CC2)=O)ccn2nncc2c1 1711,C1(NC(C=NOC)=O)(CO)CCCN(C(=O)C(c2ccnn2C)C)C1 1712,CC1(C)CCC(O)(C(N2CC(CNC(c3csc(C(F)F)n3)=O)C(O)C2)=O)CC1 1713,CC1CN(C(=O)Cc2cccnc2Cl)CC1NC(=O)C(O)C1CC1 1714,C1(N(C(=O)CC2CC2(Cl)Cl)CC)CCN(C(=O)Cc2cncnc2O)CC1 1715,CC(C)(C)C(O)C(=O)NC1CCCN(C(c2cc(F)ccc2Cl)=O)CC1 1716,c1(C(c2n(CCCC)nnn2)NCC=CC(C)(C)C)ncc(C)cc1C 1717,N1(C(CCCOCC)=O)CC2CCCC(CNC(C3CCCO3)=O)C2C1 1718,c1(NC(C2N(S(CC)(=O)=O)CCNC2)=O)sc2c(c1C(N)=O)CCOC2 1719,c1(C(=O)NC2(CF)CCN(C(C3N(C(C)=O)CSC3)=O)C2)cncc2ccsc12 1720,n1(C(C(=O)NCC2(C)CCN(C(COC)=O)C2)C)cc2ccccc2n1 1721,S(=O)(=O)(c1cc(C(N2CC=CC(NC(=O)C=CCO)C2)=O)ccc1F)NCC=C 1722,Cc1cc(C(N2CCC2C(N2CCC(O)C(C)C2)=O)=O)ccc1F 1723,N1(C(c2cc(C=C)cc(F)c2)=O)CCN(C(=O)C(C)(C)C)CC2CCCCC12 1724,N1(C(c2cn(C(C)C)nc2)=O)CCCC(C)(NC(=O)CCc2cnc[nH]2)C1 1725,c1(C(=O)NCC(CN(C(C(c2cccc(C)c2)=O)=O)C)(C)C)cc2n(n1)CCC2 1726,c1(CC)cc(C(=O)NCC(C)CNC(=O)C=CCN(C)CCOC)sc1C 1727,CCC(O)C(C)C(=O)NCC1CN(C)CCN1C(C1C=CC=CC=C1)=O 1728,N1(C(c2ccc(Cl)s2)=O)CC(CNC(C2CC(N3CCCC3)C2)=O)CC12CCC2 1729,CC(C(=O)NC1C=CCN(C(c2ccc(C3CC3)cn2)=O)C1)C(F)(F)F 1730,n1(CC(=O)NC(CN(C(=O)CCSC(F)(F)F)C)(CO)CO)cnc([N+](=O)[O-])c1 1731,C(C)(CO)(C(=O)NC1CC1NC(=O)CCc1ccccc1C)OC 1732,c1(C(N(C2CN(C(c3c(F)ccc(F)c3N)=O)C2)C)=O)cccn2c(O)nnc12 1733,c1(OC)nc(N(C)CC2CCN(C(=O)Cn3ccnc3)C2)ncc1C#N 1734,CCCC(CNC(=O)C(C)C)C(=O)NC1(C2CC2)CC1 1735,N1(C(C)C(=O)OCCSC2CCCC2)CCOCC1=O 1736,c1(CC(=O)NC2C3(CC(NC(C4N(CCC)CCC4)=O)C3)C2)cccc(F)c1F 1737,N1(CC(=O)NC2(C)CCN(C(C34CSC(C3)C4)=O)C2)C(=O)NC2(CCCC2)C1=O 1738,C1(NC(c2cc(Cl)c(Cl)[nH]2)=O)CN(C(c2cnn(CCF)c2)=O)CC2(CCC2)C1 1739,C1(CCO)CC(N=c2[nH]c(=NC3CCC(C4CC4)CC3)[nH]c3c2COC3)C1 1740,C(CC(=O)Nc1ccc(N(C)CC)cc1)(C1=CCCC1)OCC 1741,C1(CNC(C(CC#C)O)=O)CCN(C(c2scnc2CC)=O)CC1(F)F 1742,c1(C(=O)NCC(C2CCC2)NC(C(C)SC)=O)cc(C)ccc1Cl 1743,CC(C)CC(CNC(C1CCCN1C=O)=O)NC(=O)C(C)(C)COCC(F)F 1744,O(NC(=O)C(C)(C)C(C)NC(=O)C(F)C(C)(C)O)CC=C 1745,CN1CC(C(=O)NCCC2(NC(c3c[nH]c(C#N)c3)=O)CCC2)CCC1=O 1746,c1(C(=O)NC2(CNC(CCC(C)OC)=O)CCOC2)ccc(Cl)cc1O 1747,C1(C(=O)NC(c2cccnc2)C(=O)N(CCCC)C)CCN(CC)CC1 1748,c1(CN2C(CCNC(C3(C=C)CCCCC3)=O)CCCC2)ccc2c(c1)COC2 1749,C1(C(=O)NCC2(NC(c3cc(N)nc(Cl)c3)=O)CCC2)Cc2ccccc2O1 1750,[nH]1ccc2ccccc12.Cc1ccc(C(O)CNC(=O)CCn2cc(C)nn2)o1 1751,c1(C(N2C(CNC(CCC3N(C)CCC3)=O)CC2)=O)cccn2cncc12 1752,c1(C(N2C(CNC(C(CC(=C)C)C)=O)CCC2)=O)ccc2nsnc2c1 1753,C1(C)(NC(C(C2CCCCCC2)C)=O)CCN(C(c2cscn2)=O)C1 1754,CCC(C)(C)C(=O)C(=O)N1CCC(C2CCCN2C(c2ccc(Cl)o2)=O)C1 1755,c1(C(N(C2CN(C(CN(C)C)=O)C2)C)=O)cc(=O)cc[nH]1 1756,C(=O)(C1=CC2(CCOC2)C1)N1CCC(C(N(CC(CC)CC)CC)=O)CC1 1757,c1(C(N(CCNC(c2cc(OC)ncc2)=O)C2CC2)=O)ccc2occ(C)c2c1 1758,C1(C2CCCN(C(C3C(C)(C)C3(F)F)=O)C2)(NC(C=C(CCC)C)=O)CC1 1759,c1(OC)ccc([N+](=O)[O-])cc1C(N1CCN(C(=O)COc2nnc(C)s2)CC1)=O 1760,c1(C(=O)NC(C(=O)NC(CC#C)CCOC)CCC)cccc(C#N)c1C 1761,c1(CC(=O)N(C2CCN(C(C3CCCC(F)C3)=O)CC2)C)c(F)cccc1F 1762,c1(CNC2C(C(=O)NC(c3cncs3)C)CCC2)c2c(nn1C)CCC2 1763,c1(NC(C(CC)Br)=O)cc(C)cnc1COC 1764,C1(O)(CC)CCCN(C(=O)C(C)=CCNC(=O)Cn2nc(C)nc2C)C1 1765,Cc1nc2cc(C(=O)NCC(O)CN(C(=O)CC3=NNC(=O)C3)C)cc(O)c2o1 1766,CC(C(=O)N1CCC1CNC(=O)Cc1cscn1)n1ccnc1 1767,C1(C)(NC(C(C)CC2CCC2)=O)CCN(C(C2CCN(c3nccs3)CC2)=O)C1 1768,C(=O)(C(C)CCCOC)NCCCC(C)(C)NC(c1cc(CCCCC)[nH]n1)=O 1769,C#CCCCC(C)C(=O)NCC(CO)NC(c1cc(C(N)=O)[nH]n1)=O 1770,C(C(CC(=O)N1CCC(C)(N(C)C)C1)NC(=O)CC1(O)CCOC1)OC 1771,C(=O)(C1CCOc2ccc(F)cc21)N1CC(CNC(C(Br)=C(C)C)=O)C1 1772,N1(C(CC2OCC(C)(C)OC2)=O)CCCCC(NC(C2(CC3CC3)CC2)=O)CC1 1773,Cc1[nH]c(C#N)cc1C(=O)NC1(CO)CCN(C(C2CC(C)(C)CN2C)=O)C1 1774,CP(C)(=O)CCC(=O)NC1CCN(C(=O)CCCc2csc(=N)[nH]2)C1 1775,Cn1ccc2c(C(=O)NCCC3CN(C(=O)Cn4ccnn4)CCO3)ccnc12 1776,c1(SCC(=O)NCC2(COC)CN(C(C3CCC3(C)C)=O)C2)ccccc1Br 1777,c1(CC(=O)NC(CNC(c2n(CCC)ccc2)=O)C2CCC2)cnc(Cl)cc1C 1778,S1(=O)(=O)c2cccc(c2)C(=O)N1C.c1(C(CC)NCC(=O)NCC)nc(=O)o[nH]1 1779,Cc1cnn(C)c1C(=O)NCC(c1ccccc1)NC(=O)CCS(C)=O 1780,C(CCC(=O)NC(C)CN(C(=O)CCc1nc(C)no1)C)=CC 1781,C12(NC(C3ON=C(C)C3C)=O)CC(CNC(=O)CC(C)n3cccn3)(C1)OC2C 1782,C1(C(=O)NCc2ccc(C3CC3)cc2)CC12CCN(Cc1nc(C3CC3)no1)C2 1783,CS(=O)CCC(O)C(=O)NC1(C)CN(C(=O)Cc2csc(-c3ncccn3)n2)C1 1784,C1(C(=O)NC2CCOC2=O)CCCC2CN(C(=O)C3Cc4ccccc43)CC12 1785,N1(c2nnc(C34C(C)(C)C(CC3)C4)n2CCSC2CC2)CC2CS(=O)(=O)CC2C1 1786,N1(C(C2(OC)CCSC2)=O)CCCC(N(C(=O)CNS(=O)(=O)N(C)C)C)C1 1787,c1(N(CCNC(C2CC23CCOC3)=O)CC)c(Cl)cncc1[N+](=O)[O-] 1788,Cc1noc(C)c1C=CC(=O)NC1CC2CC1N(C(c1c[nH]c(C(N)=O)c1)=O)C2 1789,c1(CC(=O)NC2CCN(C(C=CC(CC)C)=O)CC2F)cn2ccccc2n1 1790,c1(OC)ccc(Cl)cc1C(=O)NC(C)CNC(=O)Cc1cccc(F)c1O 1791,CC(CC(F)(F)F)C(=O)NC(CC1CC1)C(=O)N1CC(N2CCC2)C1 1792,c1(OC)c(C(=O)NCC2CSCCS2)ccc(Cl)c1Cl 1793,C1(C(N(CCCN(CC)CC)C)=O)(COC)CCCN1C(=O)C(C)(F)F 1794,c1(CCC)cccc(C(=O)N(C)CC2COCCN2C(=O)CN(C)C(=O)OC)c1 1795,C1(CC(=O)NCCC(CNC(=O)CC(=O)Nc2nccs2)O)CC2C=CC1CC2 1796,c1(CNC(=O)OC2CN(C(=O)C3CC3)C2)ccc(I)nc1 1797,N1(C(C2C(C)(C)CCCO2)=O)CC2CCN(C(=O)C=Cc3ncc[nH]3)CC2C1 1798,CCCCC(C(=O)NC1CC2CCC1(COC(=O)C(F)(F)F)C2)CCC(=O)OC 1799,c1(NC(C2C(NC(Cn3ccc(C)n3)=O)C2)=O)ccc2c(Cl)n[nH]c2c1 1800,C(=O)(C(=O)N=S(C)(C)=O)NC(C)C(C1CCCCC1)NC(C1CC=CC(O)C1)=O 1801,C(=O)(C1SCCc2sccc21)N1C(C(C)NC(c2cc(C)ncc2)=O)CCC1 1802,c1(C(=O)NC23CC(NC(C(C(C)C)OCC)=O)(C2)C3)cc(OCC)nc(C)c1 1803,N1(C(C2(O)CCCC2)=O)CCCCC1C(=O)Nc1nccc(C(F)(F)F)n1 1804,N1(C(C=CCN(C)C)=O)CC(O)(CNC(=O)Cc2ccc(Cl)s2)C1 1805,C(C1CN(C(c2cc(C(N)=O)co2)=O)CC1C(N1CCC(C(N)=O)C1)=O)=CC 1806,c1(CC(=O)NC2CN(C(=O)C(O)CC(F)F)CC2O)cnc2ccccc2c1 1807,CC(O)C(C)(C)C(=O)NCCOCCNC(=O)C(Cl)=CCl 1808,C=CCCC(c1nnnn1C1(C)CC1)(C1CC1)NC(C)CCC=C 1809,c1(CN2CC3C(C(=O)NCCc4cscn4)C3C2)cccc2cccnc12 1810,c1(C(=O)NCC(CN(C(=O)CC2(O)CC2)C)O)n[nH]cc1-c1ccccc1 1811,c1(C(=O)NC2COCCN(Cc3cccc(OC)c3)C2)n[nH]c2cc(Br)ccc12 1812,N1(C(COCCCCC)=O)CCC(CNC(=O)C=CI)C(C)C1 1813,C1(NC(C(C)(C)c2ccc(Cl)s2)=O)CC2CC(NC(C3COC(=O)O3)=O)CC2C1 1814,C1(C(=O)NC2C=CC(CC(=O)NC(C)C(C)(C)C#N)C2)CC2CC(=O)C1O2 1815,c1(N2CC(C)C(NC(=O)C(C)(C)F)CC2)ncnc2c1nnn2CC1CC1 1816,C1(NC(COCCCC#C)=O)CC2(C1)CC2NC(=O)CCCOC1CCCCC1 1817,c1(CC)ccc(C=CC(N2CCCC2CN(C(=O)Cc2ncc(C)o2)C)=O)cc1 1818,N1(C(c2cc(OC)n[nH]2)=O)CCC(C)(CNC(C2CCC(=O)CC2C)=O)CC1 1819,C(=O)(C(C(C)C)N(C)C)NC1CC(C(N2C(C(=O)NC(C)C)CCC2)=O)C1 1820,C1(OC)CC(CNC(c2occc2CNC(c2nnc(C)s2)=O)=O)CC1OC 1821,Cc1cc(N2CCC(NC(C3C(F)(F)C34CCC4)=O)C2C)n2nc(C)nc2n1 1822,C1(=O)C(C(C)(C)C)CNC(=O)C2CCN1C2.c1(NC(CC)=O)ccc(C#N)o1 1823,C(=O)(C1=CC2CCC=CCCC12)N1CC(NC(C2CC(O)(CC#C)C2)=O)C1 1824,C1(CNC(c2cnc(OC)nc2)=O)COCCN(C(=O)C(C)SC(F)(F)F)C1 1825,c1(C(=O)NCC(C)(C)NC(Cc2c(C)noc2)=O)cnc2c(c1)nnn2C 1826,C1(CNC(C(CC)C)=O)COC(C)(C)CN1C(c1cnc(SC)nc1O)=O 1827,C12(OC)CCC(C(=O)NCCCNC(=O)Cc3cc(F)ccc3Cl)(CC1)C2 1828,c1(C(=O)NCCCC2(NC(c3cc(OC)n[nH]3)=O)CC2)c(C(C)C)cccc1C 1829,CC1CCCCN1C(c1cccnc1C(=O)OC(C)(C)C)=O.C12CC1C(=O)N2 1830,c1(C(=O)NCC2CC2CNC(C2CC(O)(c3ccccc3)C2)=O)ccc(O)cn1 1831,C(C(C)CC(=O)NC(CNC(=O)COC(C)(C)C(F)(F)F)C1CC1)SC 1832,C1(NC(CCc2nc(C)c(C)o2)=O)CC2CC(NC(C3OCCC3(C)C)=O)CC12 1833,C=CC(CCC)CC(=O)N(CCC)CCOCCC(=O)NCC=CCl 1834,C(CC(O)CNC(=O)C(Cn1ccnn1)NC(=O)CC1(O)CCOC1)OC 1835,Cc1ccc(CC(=O)NC2CCCC(NC(=O)CCn3cc(C)cn3)C2)c(F)c1 1836,CC(CC(=O)N(C1CCCN(C(=O)CCN2CCC2)C1)C)C(F)F 1837,c1(NC(C2CN(C(c3cnc(Cl)nc3)=O)CCC2O)=O)cc2c[nH]nc2cc1Br 1838,c1(C(C)=O)cn(CC(N2CC(C)(OCC(=O)NC3CCCCS3)C2)=O)nn1 1839,c1(OCC(=O)NC(CNC(C2(CC)CCCC2)=O)(C)C2CCC2)ccc(F)cn1 1840,c1(C(N2CCC(CCNC(=O)C=CC3CCCC3)C2)=O)cccc([N+](=O)[O-])c1O 1841,N1(C(CCc2n(C)cnn2)=O)CC2CC2(NC(=O)CCC2CCCOC2)C1 1842,c1(CC(N2C(CN(C(C(C)C3CCCC3)=O)C)CCC2)=O)cc(O)ccc1Br 1843,C1(OC)CN(C(C2(CSC)CC2)=O)CCC1NC(=O)C(O)CCSC 1844,c1(C(=O)NC(C(=O)NC2CC(CC(C)(C)C)C2)C2(O)CCC2)ccccc1 1845,Cc1nc(C(N2CC3(NC(c4cnoc4C)=O)CC2C3)=O)ccc1C#N 1846,CC1CCCCCN1C(=O)NC1CCOC1c1ccc(Cl)c(F)c1 1847,C1(C(N2C3(CN(C(C(CCC)CC)=O)C3)CC2)=O)Cc2ccccc2C(C)(C)C1 1848,Cc1cc(C(N2CCC(C(=O)NCC3CCCC3O)(CF)C2)=O)ncc1N 1849,C1(C(=O)NCC(COC)NC(C2C(CCOC)C2)=O)CCC2CC1CO2 1850,Cc1cc(C)c(CN2CC(F)CC2C(=O)Nc2cccc(F)c2CO)cc1C 1851,CCC(CO)(C(=O)N1C(C(=O)NC2CC3CC3C2)CC1C)OC 1852,Cc1cc(S(=O)(=O)NC2CC(C)(C)OC2(C)C)c(C)cc1Br 1853,CC1(CNC(=O)CCc2ncccn2)CCN(C(C2CC(n3ccnc3)C2)=O)C1 1854,C(=O)(CC1C(=O)Nc2ccccc21)NC(C)C(CO)NC(=O)Cc1csc(Cl)n1 1855,C(=O)(CC(F)(F)CS(C)(=O)=O)NCC(CNC(C(CC#C)C1CC1)=O)C 1856,N1(C(C(C=C)O)=O)CCC(C2OCCCC2NC(=O)CCc2ccccc2)CC1 1857,C12(C(N(CCCNC(C3(c4ccc(Cl)cc4)CCC3)=O)C)=O)C=CC(CC1)C2 1858,C(C)(CC(=O)N1CCCCC1CNC(=O)CCCCCF)(C(F)(F)F)N(C)C 1859,n1(C2C(C)C2)nc(-c2ccccn2)nc1C1CC(c2ccc(Cl)s2)C1 1860,c1(CC)cc(C(N2CCCC2C(N2CC(CC(=O)OC)C2)=O)=O)ccn1 1861,c1(C(N(C2C(C)CN(C(C34CC(F)(C3)C4)=O)CC2)C)=O)ccnc2cc[nH]c12 1862,Cn1cc(CNC(C2CC=CCN2C(=O)C(O)CC2CCCC2)=O)ccc1=O 1863,Cc1cnsc1C(=O)N(CC(C)C(=O)NC1CC(CF)C1)C 1864,CCCCC(CNC(C1(C(=O)N(C)C)CC1)=O)NC(=O)C(N1CCN(C)CC1)C 1865,c1(CCC(=O)N(C)CC2CC(NC(=O)Cc3cccnc3)C2)nnc(C(F)F)o1 1866,CCCC(C)CC(=O)NC1CCCC(CNC(c2c(C)nc(C)n2O)=O)C1 1867,CC1=NOC(CC=O)C1.n1(C2(C(=O)NC3CNC3)CC2)ccc(C2CC2)n1 1868,c1(CCC(N2CC(N(C(C(C)(C(C)C)OC)=O)C)C2)=O)c(C)nc(SC)nc1O 1869,c1(C(N2CCC(C)(NC(COC)=O)CC2)=O)nccc2cnn(C)c12 1870,c1(C(=O)NC23C(CN(C(C4CC(=O)N(O)C4)=O)C2)CC3)sc2sccc2c1Cl 1871,C1(NC(=O)CCNC(c2ccncc2)C)CCCN(C(=O)NCC2CCCO2)C1 1872,c1(CC)ccc(C(=O)NC(COC)C(=O)NCC(=O)NCC(F)F)o1 1873,c1(C(N2CCCC(N3CC(C)(C)C3)C2)C)ccc2ncsc2c1 1874,Cc1ccc(=O)n(CC(=O)NCC2CC2NC(=O)COC2(C)CCCC2)n1 1875,C1(NC(c2c(OC)cccn2)=O)CCCC12CN(C(=O)CC(C)c1ccco1)C2 1876,O=C(C1=CCCN(C(C2CCC2(F)F)=O)C1)NC(C(F)(F)F)C1CC1 1877,C12(C(=O)NC(C(=O)OC)C3CC3)CC1CN(C(=O)C(C)(C)CCl)C2 1878,n1(CCC(=O)NC2CC(NC(CN3CC(C)(OC)C3)=O)C2)c(C)cc(O)cc1=O 1879,c1(OC)ccc(O)cc1C(N1CC=C(CNC(C2(OC)CC2)=O)CC1)=O 1880,CC1CCN(C(C2CC2(C)C)=O)CCN1C(c1cc(C2CC2)no1)=O 1881,CN1CC(C(=O)NC(C)(C)CC=CC(=O)NCCOC2CCCC2)NC1=O 1882,c1(C(=O)NC(C(=O)OCC#N)Cc2ccccc2)noc2c1CCCCC2 1883,N1(CC(=O)Nc2ccccc2)CC2(CCC(CNC(C34CCCCC3C4)=O)O2)C1 1884,C1(NC(c2c(C)n(C(C)C)cc2)=O)CCN(C(=O)CCC2CCOC2)CC1O 1885,N1(C(c2c(CC)nc[nH]2)=O)CCCC(O)(CCNC(c2cnc(C3CC3)[nH]2)=O)C1 1886,c1(C(C(C)C)NC(=O)NCC2CS(=O)(=O)C2)ccc(Cl)cc1 1887,N1(C(CN(C2CCCC2)C)=O)CCC(NC(N2CCOCC2)=O)C(O)C1 1888,C(=O)(C(C)(C)C(C)C)NCC(N1CCN(C(C(C)=CC2CC2)=O)CC1)=O 1889,C1(NC(CNCC2C(NC(C(C)NC(C3CCC3)=O)=O)C2)=O)CCOC(=O)CC1 1890,CC1CCN(C(=O)Cn2cc(CO)nn2)CCN1C(c1ccc(C(N)=O)cc1)=O 1891,CCCC(CNC(c1ccsc1C)=O)C(=O)NCC(F)(F)C(C)(C)O 1892,c1(C(=O)NCC2COC(CNC(c3cc(Cl)no3)=O)C2)cccc(CO)n1 1893,CC(C)(C)C(=O)NCC(=O)NCC1CCCN1C(=O)Cc1ncc(Cl)s1 1894,Cc1sc(-c2nc[nH]n2)nc1C(=O)N(CCCNC(=O)CC1CCCC(C)C1)C 1895,C1(C(N2CCC(Cn3cc(CCN(C)C)nn3)CC2)=O)CC1C1CCCC1 1896,CC1CCC(NC(=O)OC(C)(C)C)CN1C(c1ccoc1I)=O 1897,c1(C(N2CCN(C(c3ccc(C)cc3)=O)C3C2C3)=O)ccnc2ccnn12 1898,c1(C(C)NC(C2CC=CC2)=O)ccc(CNC(C2(c3cccs3)CC2)=O)cc1 1899,c1(OC)ccc(C(N2CC(OC)C(NC(=O)CSC(C)C)C2)=O)c(N)c1Br 1900,C1(NC(c2cccc(OC)c2)=O)CCN(C(=O)CC(O)C2CCCC2)C1(C)C 1901,CCCC(O)CC(=O)N1CCC(C(C)(C)C)(CNC(=O)CCS(C)(=O)=O)C1 1902,CC(C)S(=O)(=O)CC(=O)N1CC(OCCC(=O)NC2CC3(C2)CC3F)C1 1903,CCC(C)(COC)CNC(C1CCN(C(=O)CCCCN(C)C)C1C)=O 1904,N1(C(C=Cc2ccc(C)o2)=O)CCCC(NC(C2(N(C)C)CCC2)=O)C1C 1905,N1(C(COCC(=C)C)=O)CCC(N(C)Cc2cncs2)CC1 1906,N1(C(c2cc(Cl)cc(Cl)c2O)=O)CCC2CCN(C(C34CCC(C3)C4)=O)CC12 1907,C1(C)(C(N(CC(CNC(c2c(C)n(C3CC3)nc2)=O)(C)C)C)=O)COC(C)CO1 1908,CC1(C)CC(NC(=O)NCC(C)(F)C(C)(C)F)c2ccccc2O1 1909,C(C)(C(=O)NCC(C)(C)CNC(=O)CC(C)C1CC1)(C(C)C)NC(C)=O 1910,C(=O)(CC(C)(O)COC)NC(CC)CNC(=O)Cc1ncccc1C 1911,n1(CC)cnc2c(NC(C)CCCO)[nH]c(=NCCCCCN3CCCC3)nc12 1912,Cc1ccc(CC(=O)NC2CCC2NC(c2cccs2)=O)s1 1913,N1(Cc2nc(CCCC)sc2)CCC(C)C(NC(C2CCS(=O)(=O)C2)=O)C1 1914,Cc1ccc(C)c(C(=O)NCC(CC(C)C)NC(c2cccnc2)=O)c1O 1915,C1(NC(CCOCC)=O)CCC2(CCN(C(c3ccsc3C#N)=O)CC2)C1 1916,c1(C(N2CCC(O)(CC(N3CCC(C#N)CC3)=O)CC2)=O)c(Cl)cc(Br)cc1Cl 1917,C(CN=c1nc(-n2ccnc2)cc[nH]1)C1N(Cc2cc(C)nc(O)c2)CCCC1 1918,C1(CNC(C(C)CN2CCCCC2)=O)(NC(=O)CCc2cc[nH]n2)CCCCC1 1919,N1(C(CC2CCN(C)CC2)=O)CC(NC(C2CC2c2ccncc2)=O)CC(O)C1 1920,c1(C(=O)NCCCN(C)C(C2CCCS2)=O)cc(S(=O)(=O)N2CCOCC2)c[nH]1 1921,C1(NC(c2c(C(N)=O)csc2)=O)CS(=O)(=O)C2CN(C(c3cnns3)=O)CC12 1922,c1(C(=O)NC2CC(CCNC(CC3(OC)CCC3)=O)C2)cncnc1C 1923,c1(CC)cnoc1C(=O)NC1CC(C)(NC(=O)C(C)C2CCCO2)C1 1924,CC1CC(CNC(C23CSC(C2)C3)=O)CN1C(=O)CC1(N2CCCC2)CC1 1925,CC(C)S(=O)(=O)c1cnc(NC(=O)Nc2ccc(CS(C)(=O)=O)cc2)nc1 1926,N1(C(C2CC2C(=O)NC2CCCOC2)C)CC(CO)C2(CC2)C1.C1(=O)CN1 1927,C(CCC(C)(C)CNC(C1CC1C(C)(C)O)=O)NC(COCCOCC)=O 1928,CC1OCCCC1C(=O)NCCCN(C1CCCC1)C(C1CSC1)=O 1929,CCC(CC)(CO)C(=O)N(C)CC1(CNC(C2CCC3CCC23)=O)CC1 1930,Cc1cnc2c(C(=O)NC(CNC(=O)C=C3CCC(C)C3)C3CC3)cccn12 1931,C1(C)(CNC(c2n(CCOCC)nnn2)c2cscc2Cl)CC2(C1)CC2(F)F 1932,N1(C(C2CCCN(C(CC3(C(=C)F)CCC3)=O)C2CC)=O)CCC(O)C(F)(F)C1 1933,C1(C)(C(=O)NC2CC3CN(C(C4(C)CC(C)OCC4)=O)CC32)CCCCC1(F)F 1934,c1(C(N(CC(C)NC(=O)CCC2CCCC2)C)=O)ccc(N)c(Cl)c1 1935,c1(C(=O)NCC2CCN(C(c3c(CCC)n(C)nc3)=O)C2)cc(Cl)ccc1OC 1936,c1(OC)ccccc1C(C)C(=O)N(C1CN(C(c2c(Cl)nsc2Cl)=O)C1)C 1937,c1(C(=O)NCCOC2CN(C(c3c(C)oc(Cl)n3)=O)C2)ccc2c(c1)CC(=O)N2 1938,c1(CN(C(CC)C)C(C2CCCC23CC3)=O)ccc(F)cc1 1939,c1(OC)ccc(O)c(C(=O)NC2CCC(NC(=O)C(CCSC)NC=O)C2)c1 1940,c1(OC)nc(C)cc2ccc(C(=O)NCC(C)NC(C3C(C)(C)C3(C)C)=O)cc12 1941,c1(C(=O)NC2CC(NC(C=CC3(C)COC3)=O)CC2O)cc2cnccc2o1 1942,C1(CN(C)C(c2ccc(C(C)(C)C)nc2)=O)CCN(C(=O)C(F)(F)CF)CC1 1943,C1(CNC(C(CSC)O)=O)CN(C(c2ccc3nccn3c2)=O)CCC12CCC2 1944,Cc1scc(C(=O)NCC(c2ccc(F)cc2)NC(c2nnsc2C)=O)c1C 1945,CC1CCC=C1C(=O)N1CCC(NC(=O)CCN2CCCC2=O)C12CC2 1946,Cc1cc(F)c(C(=O)NC2CCCCC2CNC(c2nc(O)sc2C)=O)c(Br)c1 1947,c1(C(=O)NC2CCN(C(CN(C)C)=O)CC2CO)c(F)ccc2occc12 1948,Cc1cc(C(=O)N(CC(C)NC(C23CCCC2C3)=O)C)cc(C)n1 1949,C1(NC(=O)Nc2cccc(C3CC3)c2)C2Cc3cc(Br)ccc3C12 1950,c1(OC)ccnc(O)c1C(=O)NCC(C)N(C)C(c1cc(CO)[nH]n1)=O 1951,CC(C)(CCCCNC(=O)C(O)C1CC1)NC(c1cc(Cl)n[nH]1)=O 1952,C1(NC(=O)C(F)Cc2ccon2)COC2(CCN(C(=O)C=Cc3nccs3)C2)C1 1953,c1(NCC(C(C)C)OC)ccc(S(=O)(=O)N(C)Cc2ccnc(SC)c2)c(Cl)c1 1954,C1(C(=O)NC(C)CC(N)=O)N(C(C2CN3CCC2C3)=O)CCCC1(C)C 1955,c1(C(N2C(C)(CNC(=O)C(F)CC3CC3)CCC2)=O)cccc2c1NCCC2 1956,N#Cc1sc(=NC2(C3CN(C(=O)CCNCS(=O)(=O)C(F)(F)F)CC3)CC2)[nH]c1Cl 1957,c1(C(N(CCCNC(C=C(C)C)=O)C(C)C)=O)nncn1C1CC1 1958,C1(OC)(CNC(=O)CC2CC3(CC3)CO2)CCN(C(C2C(C)(C)C2(F)F)=O)CC1 1959,C1(CCNC(=O)C(O)C2CC2)CCCCN1C(C1CCC(O)CC1)=O 1960,c1(NC(N2CCC(CN(CC(CC)CC)C)CC2)=O)c(Br)ccc(C)c1F 1961,S(=O)(=O)(c1ccc(NCCc2cnoc2)cc1Cl)NC(c1ccn(C2CC2)n1)C 1962,C1(NC(C2C(CC)C2)=O)CCN(C(=O)C(Cc2ccccc2)N(C)C)CC1(C)C 1963,c1(C(=O)NCC2CN(C(C3COCC3C(F)F)=O)C2)ccc(-n2cccn2)cc1 1964,N1(C(Cc2cc(C(C)=O)sc2)=O)CCN(C(c2cnnc(O)c2)=O)C(CCO)C1 1965,C1(C(N2CCC(Cc3cn(CC(CC)O)nn3)CC2)=O)CCc2ccccc2C1 1966,C1(C(N2CC3CN(C(CC(C)C)=O)CC3C2)=O)CCc2nn(C)cc2C1 1967,C(=O)(C(C)(CC)CO)NCC(N1CCN(C(C2C(CN(CC)CC)C2)=O)CC1)C(F)F 1968,C(CCN=C(NCCCOC(C)(C)C)NC(C1CCOC1)C)NCC(C)C 1969,N1(C(CC2(OC)CCCC2)=O)CC2CCCC1C2CNC(=O)CSC(F)F 1970,CC1(C)CN(C(c2cccnc2)=O)CC(CNC(=O)Cc2ccc(F)cc2Cl)O1 1971,Cc1cnc(NCCC2CCS(=O)(=O)C2)c(S(=O)(=O)NCCCCCF)c1 1972,C1(NC(C(COC)(C)C)=O)CCN(C(=O)C(C)OCC(C)C)C12CC2 1973,N1(C(C2(C(F)(F)F)CC=CCO2)=O)CCN(c2ccccc2OC(F)F)CC1 1974,c1(C(=O)NCC2CCN(C(C3CN(CCC)C(=O)C3)=O)CC2)cc(C#N)[nH]c1C 1975,C(CC(=O)N1CC2(CCCC2)C1)(C(F)(F)F)NC(=O)C=CC1CCOCC1 1976,c1(NC(N2C(C)CN(Cc3ccc(Cl)c(Cl)c3)CC2)=O)cn2cccnc2n1 1977,C=C(C)CCCC(=O)NC(C)Cn1cc(CN(CC)CC)nn1 1978,N1(C(CCC(=O)OC)=O)CC2(NC(=O)CN(C3CCSC3)C)CCCC2(F)C1 1979,C1(NC(CC(C=C)C)=O)CC2CC1N(C(c1cnc(C(C)(C)C)o1)=O)C2 1980,CN(CCc1cccc(Br)c1)N1CCCC(OC(C)(C)C)C(O)C1 1981,C12(C(N3CC(CCNC(C4CNC(=O)N4)=O)C3)=O)CCCC(CCC1)C2O 1982,CCCCC(O)CC(=O)NC1CCCN(C(=O)C(C)(C)C(C)C)CC1 1983,C12(C(=O)NC(C(C)C(=O)N(CCC(O)CO)C)C)CCC(CC1F)C2 1984,N1(C(C2C(C=C)C2)=O)CC2CCC1CN2C(=O)CNC(=O)OC 1985,N1(C(Cc2n(C)nnc2)=O)CCC(CNC(C2CNC(=O)C2)=O)C12CC2 1986,C1(C(=O)NC2C(CNC(c3sc(CCC)c(COC)c3)=O)C2)C(C2CC2)C1(F)F 1987,N1(C(CCC)=O)CC(C(=O)NCc2nnc(C)s2)C(F)(F)C1 1988,C=CCCCCCCC(=O)NC1CCCCN(C(=O)C(C)C(O)CC)C1 1989,N1(C(C2(C)CC2)C)CCCCC(Nc2cc(C(F)(F)F)ncn2)C1 1990,C1(C(N2CCC(NC(Cc3scc(C)c3)=O)C(CO)C2)=O)C2(CCC2)C12CCC2 1991,n1(C(C)C)cc(CC(=O)NC2CCCC2NC(=O)CCOC2CCCCC2)nn1 1992,c1(C(=O)NC(C2CCOC2)CNC(=O)Cn2ccnn2)ccc(O)c(Br)c1 1993,C1(NC(C(C#C)(C)C)=O)CC2CCC1CN(C(C1CCC(F)CC1)=O)C2 1994,c1(C(=O)NCCC2(O)CCN(C(C34OC(C)C(C3)C4)=O)C2)cccc2occc12 1995,C1(c2nnnn2CCCF)(NCc2ccc(CCC)s2)CSC(C(C)(C)C)C1 1996,n1(CCCC)ncc(C(N2CC(NC(=O)CC(CC)C3CC3)C(C)C2)=O)c1C 1997,c1(C(=O)NCC(C2CCC2)NC(c2csc(Cl)n2)=O)ccc([N+](=O)[O-])cn1 1998,C12(NC(C3CC3[N+](=O)[O-])=O)CCC(C1)N(C(=O)CNc1ccc(C(F)(F)F)cn1)C2 1999,C12(CNC(CC(=O)OCCC(C)C)=O)CN(C(=O)C=CC3CCC3)CC1CCO2 2000,N1(C(CC2N(C(CC(C)C(F)F)=O)C3C2CCC3)=O)CCC2(CCC(O)C2)C1 2001,C1(CNC(C2CCC(CC)O2)=O)(OC)CCN(C(=O)C(F)(F)C2CCCC2)C1 2002,Cc1ncnc(C)c1CC(=O)NCCCNC(C1CC2(F)CC1C2)=O 2003,c1(CC(=O)NC(CC=C)CNC(=O)C(C)O)ccc(Cl)nc1F 2004,Nc1c(C(N2CCC(CNC(c3ccc(CF)cc3)=O)CC2)=O)ccc(Cl)c1Cl 2005,C1(CNC(CSC(C)C)=O)CCN(C(=O)CN2CCC(C)C2)C1 2006,C1(CC(=O)N(CCn2cc(-c3ccncc3)nn2)CC2(O)CC2)CC2COCC12 2007,N1(C(C2C3(CCN(C(C4(CC)CCC4)=O)C3)C2)=O)CCC(C2(C)CC2)CC1 2008,c1(C(N(C2CCN(C(=O)Cc3ccco3)C2)CCC)=O)ccc(C(N)=O)[nH]1 2009,N1(C(C2C(CC)CCN2C(c2cc(C3CC3)[nH]n2)=O)=O)CCc2oc(C)nc2C1 2010,C1(CC)CN(C(C2(C3CC3)CC2)=O)CCC1NC(=O)C(C#N)=CC(C)C 2011,c1(OCC(C)C)ccccc1C(=O)NCCC(C)(C)NC(=O)Cc1ccsc1Cl 2012,CCC(CC)(C(=O)N(C)CC1(CNC(C2CC(OCC)C2)=O)CC1)OC 2013,C1(NC(C(c2ccnn2C)C)=O)CCOCC1C(=O)N(C)Cc1cccnc1O 2014,C(=O)(CCC(C)(C)c1nn[nH]n1)N(C(c1ccc(F)cc1)(C)C(=O)O)C 2015,C(=O)(C(O)C1=CCCCC1)NC(C(=O)NC(CCC(C)C)C)C1CC1 2016,N1(C(CC2COCC(C)O2)=O)CC(C(=O)N(C2CN(C)C2)C)C(C)(C)C1 2017,c1(CC)cccc2c1CN(C(=O)C(=O)Nc1ccc(Cl)cc1)CC2 2018,c1(NC2C(NC(c3cccc4nc(O)[nH]c34)=O)CC2)ncc(Cl)cc1[N+](=O)[O-] 2019,CCCC(O)CC(=O)NC(CNC(c1cc(N2CCCC2)ncn1)=O)CCOC 2020,Cc1cccn2cc(C(=O)NC3(C)CC(NC(=O)C(O)P(C)(C)=O)C3)cc12 2021,C(=O)(C(C)C(CC)CC)N1CC(CN(ONC(=O)OC)C(C)(C)C)C2(C1)CC2.CC 2022,c1(C(N(C(C)CN(C)C(C2C(C)C2C)=O)C)=O)ccc(-c2ccccc2)o1 2023,c1(NC(C2(NC(C3CC(Cl)(Cl)C3)=O)CCSC2)=O)cccc(F)c1 2024,C=C=C(C)CC(=O)NC(C(=O)NCCC1CC2C=CC1C2)c1cccs1 2025,CC(N=c1ccnc(Cl)[nH]1)C1CCN(C(=O)C(C)Cc2ccccc2)C1 2026,C1(C(N2CCC(NC(c3c(C)ocn3)=O)C(O)C2)=O)CCc2ccc(F)cc2C1 2027,c1(C(N2CCC(N(C(c3cc(C)cc(O)n3)=O)C)C2)=O)ccc2c(c1)N(C)CC2 2028,Cn1cc(C(N)=O)c(=NC(=O)C2CC(NS(=O)(=O)c3ccc(Cl)cc3)C2)[nH]1 2029,C1(OC)(CNC(=O)Cn2cc(Br)cn2)CCN(C(C23COCC2C3)=O)CC1 2030,C1(C(=O)NC(c2nccc(O)n2)C)C=CCN(C(=O)Cn2ccnc2)C1 2031,C=CCCC(F)(F)C(=O)NC1CN(C(c2cc3ccccc3s2)=O)C1 2032,Cc1nc2cc(C(=O)NC(C)CCNC(C3CC(C)CC(=O)N3)=O)[nH]c2s1 2033,C(C(C)C(=O)NCCCC1(NC(C2CCC(=O)C2)=O)CC1)OC 2034,C1(C(=O)NC(C)CNC(=O)Cn2cnnc2)CCCCC12CCC2 2035,N1(C(c2c(C)noc2N)=O)CCCC(C)(C(=O)NCC2(C)CSC2)C1 2036,C1(CNC(c2nocc2Cl)=O)CCN(C(=O)CCn2cc([N+](=O)[O-])cn2)C12CC2 2037,c1(C(N(C2(C(N(CC(C)(C)O)CCC)=O)CC2)C)=O)cnn(C)c1Cl 2038,C1(NC(C(C(COC)C)C)=O)CCCC12CCN(C(=O)Cn1nnc(=N)[nH]1)CC2 2039,C1(C(N(C)CC2COCCN2C(c2n[nH]cc2Br)=O)=O)CCC2(CCC2)O1 2040,c1(CCCC)ccc(C(N2CC(CNC(C3CCCOC3CC)=O)C2)=O)cc1N 2041,C1(NC(C2C(C(=O)OC)C=C2)=O)CCN(C(=O)C(C)OCC(C)C)CC1OC 2042,C1(C(=O)NCC2CCCC(CNC(=O)CCF)C2)CN2CCCC1C2 2043,c1(N2C(C)C(N(C)C)CC2)ccc(S(=O)(=O)NCCCc2cnoc2)cn1 2044,C1(C(N(CCC(=O)Nc2cnsc2)C2CC2)=O)C=CCCC1 2045,c1(OC)ccc(C(=O)NCCNC(C2CCCN(C(C3CC3[N+](=O)[O-])=O)C2)=O)cc1 2046,c1(OCC)c(Cl)cc(NC(c2ccc([N+](=O)[O-])o2)=O)cc1Cl 2047,O=S(=O)(c1cncc(Br)c1)NC1CCC(NCc2ccc(Br)cc2O)C1 2048,N1(C(C2CCN(C)CC2)=O)CCC(NC(=O)CO)C(F)(F)CC1 2049,N1(C(C(C)(C)c2cscn2)=O)CCC2(CCC2NC(=O)C=Cc2cccs2)CC1 2050,c1(CC(=O)N(CCCNC(C(C)C2CCC2)=O)C)ccc(Cl)c2cccnc12 2051,N1(C(CC(C)(C)O)=O)CCN(C(=O)C=Cc2ccccn2)CC1CS(C)(=O)=O 2052,C1(CNC(=O)COc2ccccc2)CCC(NC(C2CC2C2CC2)=O)CC1 2053,CCCC(C)CC(=O)N(C1CCCN(C(c2sc(N(C)C)nc2C)=O)C1)CCF 2054,C1(CNC(c2cc(C)sn2)=O)CCCCN(C(c2cc3[nH]ccc3s2)=O)C1 2055,c1(CC(=O)NCCNC(c2c(Cl)csc2Cl)=O)ccc2cccnc2c1 2056,c1(C(=O)NCCSCCC(F)(F)F)cnc2c(Br)cc(Br)cc2c1 2057,C1(C(=O)NC(c2cccc(C)n2)CC)CCCN(C(=O)C(=O)N(C)C)C1 2058,C(CC1=CCCCC1)N(C(c1c(C)occ1)C(=O)NCc1nnn(C)n1)C 2059,N1(C(CCCOCCC)=O)CCCC2CN(C(C3(F)CC34CCCCC4)=O)CC12 2060,c1(C(=O)NCCCCCNC(c2c[nH]c(=O)cn2)=O)cccc2cnccc12 2061,C=CCC(CNC(c1ccn(CCOC)c1)c1nnnn1C)CC(C)C 2062,C(=O)(CS(=O)(=O)C1CC1)NCCC1CC(NC(c2c(NCC)c(F)ccc2)=O)C1 2063,C1(CC)CCCN(C(c2ccc(OC)s2)=O)C1C(=O)NC(C12CCC(CO1)C2)C 2064,c1(CCC)c(C(N2CC(O)(C(C)NC(=O)CNS(=O)(=O)CC)C2)=O)nnn1CC 2065,c1(CC)nnsc1C(=O)NC1CN(C(=O)CCc2ncccn2)C1 2066,c1(C(=O)NC2C3CC(NC(C4C(C)CCO4)=O)CC32)ccc2[nH]ccc2c1 2067,C12(NC(c3cnns3)=O)CCN(C(=O)CCc3cncc(Br)c3)CC1C2 2068,N1(C(c2nn(CC)c(C)c2)=O)CCN(C(=O)C=CCO)CC1CC(C)(C)C 2069,c12c(Cl)ccc-1c2F.N1(C(c2cc(Br)c[nH]2)=O)CCN(c2ccnc(O)c2)CC1 2070,c12cnc(cc1C(F)F)Oc1ccc(cc1)CNC2=O.N1(C(C)=O)CCOC2CC12 2071,N1(C(C(CC)SC)=O)CCN(C(=O)CCCn2cncn2)CC1COC 2072,C=CCC(CC)C(=O)NCC1CN(C(c2nnn(C(C)C)c2C)=O)CCN1C 2073,c1(C(N2CCC(CNC(C3CN4CCC3C4)=O)C2)=O)cn2ccccc2n1 2074,C1(C(=O)NC(CN(C(C2(C)ON=C(C)C2)=O)C)(CO)CO)CC2CC1CC2O 2075,CS(=O)(=O)c1ccccc1C1=CCN(C(=O)CCC2CCCC(O)C2)CC1 2076,C(C(=O)NCC)(c1ccns1)N(CCCC)CCOC 2077,C1(NC(c2cc(CC)sc2)=O)C=CCN(C(=O)COc2ccccc2)C1 2078,c1(CC)ccc(N)c(C(=O)NC2CN(C(=O)C(O)CC)CCC2C(F)(F)F)c1 2079,Cn1ncnc1C(=O)NCC1OCCC1C(=O)NOCCC(F)F 2080,O(C=CC(=O)N(C1CN(C(=O)CCc2ccc(Br)s2)C1)C)CC 2081,c1(C(=O)NCC(CO)NC(c2c(C)nn(C(C)(C)C)c2)=O)ccc(N=[N+]=[N-])cc1 2082,C=Cc1cnn(C)c1C(N1CCC(N(C(c2cc(OC)ccc2F)=O)CC)C1)=O 2083,C1(CNC(=O)NCCS(N)(=O)=O)(Cc2nccc(C(F)(F)F)n2)CC2(CCC2)C1 2084,N1(C(C2(OC)CCOC2)=O)CC2=C(C1)CN(C(c1cscc1Br)=O)C2 2085,N1(N(c2cc(C)[nH]n2)CC(N2COCCC2C)=O)CCC(O)C(C)C1 2086,C1(N(C(C(C)Oc2ccccn2)=O)C)CCCCC1NC(=O)Cc1nnc(O)s1 2087,N(C1CCCOc2c(Br)cccc21)CC#CC(OCC)OCC 2088,C12(CC(=O)NCC3(F)CN(C(C4C(C)C4)=O)C3)CCCN1CCC2 2089,C(C(C)(C)C)CCN(CCC)CN.C(CCC1CCC1)NC(=O)OC 2090,c1(C(CC(N2CCC(N(C(C3CN(C4COC4)C3)=O)CC)C2)=O)C)c(C)noc1C 2091,n1(CC(=O)NC2CCn3nnnc3C2)nc2ccccn2c1=O 2092,c1(C(=O)NCC(CN(C(=O)COc2ccsc2)CC)O)cc(C)n(C2CC2)c1C 2093,c1(C(C)C)nccc(C(N2CC3C(NC(=O)CCCc4cccs4)C3C2)=O)n1 2094,c1(COC)cccc(S(=O)(=O)NC(CCc2ccccc2)C(F)F)c1 2095,c1(C(N2C(CNC(CCC#C)=O)C(C)CC2)=O)cnc2sc(C)nc2c1 2096,CCCC(CC(=O)N1CCC(C(N)=O)(OC)C1)NC(C1(n2nccn2)CC1)=O 2097,Cc1cc(C(N2CC3CC(C(N4CCOC(CN=[N+]=[N-])C4)=O)(C3)C2)=O)cc(O)c1 2098,Cc1nccnc1C(=O)NC1CN(C(C2(OCc3ccccc3)CC2)=O)CC1C 2099,c1(C(N2CCC(C#N)(NC(C3CCNC(=O)C3)=O)C2)=O)cc(O)c(O)c(O)c1 2100,CC1CC2N(C1)C2=O.c1(CC(=O)NCCC(=O)OC(C)(C)C)ccc(F)cc1 2101,C1(NC(C(C=C)O)=O)CN(C(=O)CCc2cn(C)nc2C)C2(CCOCC2)C1 2102,C1(NC(C2N(C(=O)OCC)C(CO)CC2)=O)CCN(C)C(=O)C1 2103,CCCCC(O)C(C)C(=O)N(C(C)C(=O)NCCOC1(C)CCC1)C1CC1 2104,c1(-c2ccnc(N3CCC(O)C(C)C3)n2)c(C(C)=O)nc2ccccn12 2105,c1(C(N2CCC3(NC(=O)Cc4cnsc4)C(C2)C3)=O)ccc2sccc2c1 2106,CCCCC(C)C(=O)NCc1csc(C(=O)NC(c2ccc(O)cc2)C)c1 2107,c1(C(=O)NCC2C(NC(CC(C)F)=O)CC2)ccc(N2CCCC2)cn1 2108,Cc1c(C(=O)NC2CC(NC(c3cc(Cl)cc(Cl)c3)=O)C2)c[nH]c2nccc1-2 2109,Cc1ccc(OC(C)C(=O)NCC2CC(F)CN2C(=O)CC=C(Cl)Cl)cc1 2110,c1(C(=O)NC)cn(CC(=O)NCCCNC(=O)CC2(OC)CC2)nn1 2111,c1(CC)ccc(C(=O)NC2(C)CCCN(C(c3ccnc(C)c3Cl)=O)C2)c(F)c1 2112,C(=O)(CC(C)CC(F)(F)F)NCC1CN(C(CC2(CSC)CC2)=O)C1 2113,c1(CC)ccc(Br)cc1C(=O)NC1CCCC1CO.N12CCC(CC1)CC2=O 2114,C(=O)(C(F)C1=CCCCC1)NC1C2CN(c3nnc(C(N)=O)s3)CC21 2115,C12(COC)CCC(C(N3CCC(CNC(=O)CC(C)(F)F)C3)=O)(CO1)C2 2116,N1(C(CSc2n(C)c(S)nn2)=O)CCCC(S(=O)(=O)N(C)C)C1 2117,C1(NC(c2cc(Cl)ncc2O)=O)CCC2CCN(C(c3ccc(=O)oc3)=O)C12 2118,c1(CN2CCN(CCNC(CCC#C)=O)CC2)ccc(S(N)(=O)=O)cc1Cl 2119,C#Cc1ccc(NC(=O)C(C)(C)C2CCN(C(=O)CCOCC)C2)cn1 2120,N1(C(C2(C)ON=C(C)C2)=O)CCN(C(c2cc(N)c(Cl)c(O)c2)=O)CC(C)(F)C1 2121,N1(C(c2c(COC)ncs2)=O)CC(NC(c2cnn(C)c2C)=O)CC1C 2122,C12(CNC(C(C)C3CCC3)=O)CCCC1CN(C(c1cnc3[nH]ncc3c1)=O)C2 2123,c1(C(=O)NC(CC2CN(C(C3(CCOC)CC3)=O)C2)C)ccc(O)nc1 2124,Cc1cc(NC(C2CC2NC(c2cc(Cl)ccc2O)=O)=O)ncc1F 2125,C(=O)(C1c2c[nH]nc2CCC1C)N1CC(CNC(Cc2ccc(C)s2)=O)OCC1 2126,Cc1ccccc1OCCC(=O)NCC1CC(F)CN1C(=O)CC(F)(F)Cl 2127,N1(C(C2CN(CC)C(=O)N2)=O)CCN(C(c2cc(C)cs2)=O)C2COCC12 2128,C(CC(F)F)(C(=O)NCC1(O)CCN(C)C1)N(C(c1n(CC)ccc1)=O)C 2129,C1(CNC(C2(OC)CCOC2)=O)CN(C(=O)CC2(C)OCCO2)CCC1(C)C 2130,C(CCCCC(=O)NC1CCCC(CC)C1)=CCCC 2131,C1(NC(=O)CC2CCCC2NC(C23CC2CNC3=O)=O)CCC=CCCC1 2132,c1(C(=O)NC(C)CCC(=O)NCCOC2(C)CCC2)c[nH]c2ncccc12 2133,c1(C(=O)NCC2(C)CCCN(C(C3(C)CNC(=O)C3)=O)C2)cccn2nnnc12 2134,c1(-c2cccc(CN(C3CCCCC3)CC(C)C)c2)ccn(C)c(=O)c1 2135,N1(C(c2n(C)ncc2)=O)CCC2CCN(C(c3n[nH]c(C4CC4)c3Cl)=O)CC12 2136,C12(C(=O)NC(COCCOC)C)CC(NC(=O)CC3CCSC3)(C1)C2 2137,c1(C(=O)NC2CC3(C(C(N(C4CC(=C)C4)C)=O)C3)C2)ccc(C#N)cn1 2138,N1(C(C(C=CCCC)O)=O)CCCCC(NC(c2ccc(SCCC)cc2)=O)C1 2139,CCC(C)(COC)C(=O)NC(C(=O)N(C)CC1(COC)CCC1)C(C)C 2140,C(=O)(C1=CSCS1)N(CCCCN(C(=O)C=Cc1ncc[nH]1)C)C 2141,C1(NC(C2CCO2)=O)(CO)CCN(C(c2ccc(SC(F)(F)F)cc2)=O)C1 2142,c1(C(N2CCN(C(C#CC3(CC)CC3)=O)CC2)=O)cccc2cc(F)ccc12 2143,N1(C(c2cn(CC(N)=O)nn2)=O)CCCC(N(CCO)C(c2cnccn2)=O)C1 2144,Cc1nn(CC(=O)NC(C)CNC(=O)Cc2ncc(Cl)s2)c2ncccc12 2145,CC(F)CC(=O)N1CCC(NC(=O)Cc2cc[nH]n2)C1 2146,c1(OC(C)C(N2CCCCC2CNC(c2ccc(Cl)cn2)=O)=O)ccccc1F 2147,n1(CCSC)nnnc1C(c1csc(-c2ccsc2)n1)Nc1nccn1C 2148,c1(C(=O)NC2CCN(C(C3CCC(CC)CC3)=O)C2)nn(C)c2ccc(Br)cc12 2149,N1(C(CCc2n(C)cnn2)=O)CCC2(COCC(CNC(C3(CO)CC3)=O)O2)C1 2150,c1(OC)ncc(C(=O)NCC2CCN(C(C3CC(F)C3)=O)C2)cn1 2151,c1(C(=O)NCC(c2ccccc2)NC(C2(CC=C)COC2)=O)ccc(N)c(N)n1 2152,c1(OC)c(N2CCOC(C)(CNC(C3(C(=O)N(C)C)CCC3)=O)C2)ncnc1C 2153,Cc1cc(CC(=O)NC2CN(C(c3cn[nH]c3C(C)C)=O)CC2(C)C)cc(F)c1 2154,CC(O)CCC(=O)NCC(C)N(C(=O)CCc1ccco1)C 2155,Cc1ncc(Cl)cc1C(N1CCC(O)(C(F)(F)C(N)=O)C1)=O 2156,CS(=O)(=O)c1cnn(CC(=O)NCC2OCCC2C(=O)O)c1 2157,C(=O)(CN1C(=O)C(NCC2CCCN2C)CCc2ccccc21)NC(C#C)C 2158,N1(C(c2c(C)cccc2Cl)=O)CCOCC12COCCN(C(C1CCOC1)=O)C2 2159,c1(C(N(CC(C)N(C(=O)CCc2ccon2)C)C)=O)ccc(S(N)(=O)=O)o1 2160,C1(C(C)NC(C2(N(C)C)CCCC2)=O)CCN(C(=O)CN(S(C)(=O)=O)C)CC1 2161,c1(C(N2CC3C(NC(C4CCC(OC)C4)=O)C(C3)C2)=O)cccc(C)c1[N+](=O)[O-] 2162,C(=O)(CC(F)(F)F)NCC1C(NC(C2(CC#C)CCCO2)=O)CC1 2163,N1(C(C2N(C(C)=O)CCC2)=O)CCC(CNC(C2(C)CC2(F)F)=O)CC1 2164,C1(OC)(OC)CCC1C(=O)N(CC(=O)NCc1ccoc1)C(C)C.C1CC1 2165,N1(C(c2cc(CCC)on2)=O)CCC(NC(C2CC(CCC)C2)=O)CC(C)(C)C1 2166,c1(N2CCCC(N(C(COCc3cc(C)on3)=O)C)C2)ncc(Br)cc1C#N 2167,N1(C(CCNC(COC)=O)=O)CCCC(C)(C)C1C(N1CC(c2nn[nH]n2)C1)=O 2168,c1(C(N(C(CC)C(=O)N(C2(C)CC2)C)C)=O)ccc2n[nH]cc2c1 2169,N1(C(CCc2cc(C)no2)=O)CC2C(NCc3ccn(C(C)C)n3)C2C1 2170,c1(NC2CN(C(C)=O)C2)ncccc1S(=O)(=O)N1CCC(=C(F)F)CC1 2171,C1(C(=O)NCC(CCOC)NC(c2nocc2Br)=O)CC1C1CCC1 2172,C1(C(=O)NCCC(CNC(c2c(C)ccs2)=O)O)Cc2c(F)cccc2O1 2173,N1(C(C2(C(=O)O)CCCC2O)=O)CCS(=O)(=O)CC1C1CC1 2174,N1(C(Cn2c(CCC)ncc2)=O)CCOCC1CNC(C1C=CCS1)=O 2175,c1(C(=O)NCC(CCC)NC(=O)CCc2nc(CC)no2)ccc(CCF)cc1 2176,c1(C(=O)OC)c(C)[nH]c(C(=O)NCCN(C)C(c2c[nH]nc2S(N)(=O)=O)=O)c1C 2177,N1(C(=O)Nc2ccc(C(=O)OC)c(Cl)c2)Cc2cccc(Cl)c2C1 2178,c1(CC)cc(Br)ccc1CN1CC(C(=O)NCc2ccnc(Br)c2)CC(F)C1 2179,C1(NC(C2(NC(c3cccc(=O)n3C)=O)CCN(C)C2)=O)CN2CCC1(F)CC2 2180,C1(O)(CC(N2C(Cn3cc(C(C)(C)OC)nn3)CCC2)=O)CCN(C)CC1 2181,c1(SCC=C)cccc(C(=O)NCCOCCN(C(=O)C(C)=C2CCC2)C)c1 2182,C1(CN(C(=O)C(=O)NC2CCCC(C(F)(F)F)C2)C)CC(=O)NC(=O)C1 2183,C1(NC(C2CC(O)(CNC(C(C(C)C)=O)=O)C2)=O)C=CC(C)(C)CC1 2184,c1(-n2c(CCCCCOC)nc(CCOC)n2)cc(C)ccc1C 2185,C1(CC=C)(C(=O)NCC(CCC)OC)CCCN(C(c2cnc(=N)[nH]c2)=O)C1 2186,C(=O)(C(C)(C)C(C)NC(c1cc2n(n1)CCC2)=O)NCC(CC)(C)OC 2187,C1(C(N(CC(O)CNC(C2(Br)CC2)=O)C)=O)CC12CCOCC2 2188,N1(C(C(CN(C)C)NC(=O)C(=Cc2cccnc2)F)=O)CC2(CCC(=O)O2)C1 2189,CCC(Cc1ccccc1C)C(=O)NCC(C)(O)CNC(C1(C(C)(F)F)CC1)=O 2190,C12(NC(C(CSC)OC)=O)CCCC1(F)CN(C(=O)CCCC(F)(F)F)C2 2191,N1(C(CCOC)=O)CC(C)CN(C(c2ccc(-c3ccc(F)cc3)o2)=O)C(C)C1 2192,N1(C(c2ccc(OC)cc2)=O)CCC(F)CC1C(=O)Nc1cc(C)cc(O)c1 2193,c1(OCC)nccc(C)c1NC(c1ccc(-c2c[nH]c(=N)c(C)c2)c(C)n1)=O 2194,C(=O)(CC(C)C(C)(C)C)N1CC(C=CC)C(C(=O)NC2CN(CCC)C2)C1 2195,c1(-n2cc(C3CCN(C(=O)Cc4cc[nH]c4)C3)nn2)cncc(Cl)c1 2196,c1(OC)ccc(C)c(C(N2CCC(C(C)NC(=O)CCN(C)C(C)=O)C2)=O)c1N 2197,C1(C(=O)NC2CC(CF)C2)C2CC(O)C(C2)N1C(c1ccn2ccnc2c1)=O 2198,Cc1cc(C(N2CCOCC(NC(c3ccc(C(F)(F)F)o3)=O)C2)=O)nc(C)c1 2199,CCCCCC(C)CC(=O)NC1CN(C(C2CC(F)(F)C2)=O)CC1SC 2200,C1(C(=O)NOCCC)(CC#C)CCN(C(c2c[nH]c(=O)cn2)=O)C1 2201,CCC(C(=O)NCc1cn(CC(C)NC(=O)C(F)C2CCC2)nn1)SC 2202,c1(SCC(N2C(C(=O)NCc3cn(C(C)C)nn3)CCC2)=O)ccccc1Cl 2203,c1(C(=O)NCC2(NC(C3CCCCC3F)=O)CC2)c(F)ccc(F)c1Cl 2204,C1(NC(C2CCCC2C(F)F)=O)CC2CC1N(C(c1ccncc1)=O)C2 2205,c1(CC)onc(C)c1CNC(=O)CCC1CCN(C(=O)CC2CCCC2)CC1 2206,Cc1c(C(=O)NCCCn2cc(Br)ccc2=O)cccc1Cl 2207,Cc1nc(C(N2CC(NC(c3cc(F)ncc3Br)=O)C(C)C2)=O)ccc1F 2208,C1(NC(COCS(C)=O)=O)CC(NC(=O)Cc2nn(C)cc2Cl)C12CCC2 2209,N1(C(CCN(CCC)C)=O)CC(S(=O)(=O)N2CCC(CCO)CC2)C1 2210,c1(C(=O)NC2C(CNC(C(CC#C)O)=O)C2)ccc(COC)c(F)c1 2211,C1(C(=O)O)(NC(C2(N)C(C(C)C)C2)=O)CCOc2ccccc21 2212,c1(CC)cnc(O)c(C(=O)N(C)CC2(O)CCN(C(=O)Cn3cnc(=N)[nH]3)C2)c1 2213,c1(OC)cccc(C(=O)NC(C2(O)CN(C(=O)CC3CCC4CC34)C2)C)c1C 2214,C(=O)(CC(C)CC)NC1(C(=O)NC(C(=O)N(CC)CC)C)CC1 2215,c1(CCNC(C2(NC(C3CCCC3)=O)CC2)=O)cccc(F)c1F 2216,c1(N(CCCS(C)(=O)=O)C)ccc(S(=O)(=O)N2CCSC3CCC23)cn1 2217,CC1CN(C(c2ccn(CC(F)F)n2)=O)CC1NC(C1CCC1(C)C)=O 2218,N1(Cc2ccc(OC)c(O)c2)CC2CCN(C(c3occc3C)=O)C2C1 2219,N1(C(C(C2CCC2)OC)=O)CC2(CC2)CC1CNC(=O)CCOCCN(C)C 2220,C1(CNC(c2c(OCC)scc2)=O)CCC(C)(C)CN1C(=O)C(C)CF 2221,c1(C(=O)NCC(C2CC2)NC(c2c[nH]cc2Br)=O)ccc(C(F)F)c(F)c1 2222,N1(C(c2ncn(CC)c2)=O)CC(C(N2CC(NC(C)=O)C2)=O)C(C2CC2)C1 2223,C(C)(CCC(=O)NCCC1(C(N2CCC(O)(C(N)=O)C2)=O)CC(O)C1)OCC 2224,N1(C(c2cncc(OC)c2)=O)CCOCC12COCCN(C(=O)C(C)C(C)C)C2 2225,N1(C(C(C)(Cl)Cl)=O)CC2CCN(C(=O)CS(=O)(=O)C(C)(C)C)CC2C1 2226,c1(NC(c2ccc(C)nc2)=O)ccc2nc(C3CC3)oc2c1.C12CC1CNC2=O 2227,N1(C(C=C(CCC)C)=O)CCN(C(=O)CC2COCC2O)CC1COC 2228,c1(C(=O)NCC(CC(=O)N(CCOC)CCSC)OC)ccc2[nH]ccc2n1 2229,C=CCCC(F)(F)C(=O)N1CC(NC(=O)C(C)=C2CCC2)C(c2ccccc2)C1 2230,N1(C(C(C(C)C)O)=O)CCC(C)(C)C1CC(=O)NCC1CCCSC1 2231,C1(CC)OCCC1C(=O)NCc1cc(C(=O)NCC2(CF)CC2)on1 2232,c1(C(=O)NC(C)C(CO)NC(=O)CCC2CC2CC2CC2)cc2n(c1)CCCC2 2233,c1(C(=O)NC2CCN(C(c3cn(CC)nn3)=O)C2C)cc2ccc(Cl)cc2[nH]1 2234,C(=O)(CC1=CCOCC1)NCC(c1cccc(Cl)c1)NC(C(CC#C)(C)C)=O 2235,CCCN=C(NCC(C)OC(C)(C)C)NC1CC1(C)C.n1(C(C)C)cccn1 2236,C=Cc1ccc(C(N2CC3CCC2C3NC(=O)Cc2ccn(C)n2)=O)cc1 2237,C(=O)(C(O)CC(F)F)N1C(CCN(C(CCC(C)C)=O)C)CCCC1 2238,C1(CNC(Cc2c(CC)con2)=O)CN(c2cc(C)nc(SC)n2)CC(C)(C)O1 2239,c1(-c2nc(CCOC)nn2CC(C)(C)CO)cc(C)nc2c1nc(C)n2C 2240,CC(C)(CC#N)C(=O)N1CCC(NC(=O)C(c2ccccc2F)(C)F)C(O)C1 2241,Cc1cc(C(=O)NCC2CN(C(=O)CCCC(C)(F)F)CCC2C)c(N)c(Cl)c1 2242,c1(C(=O)NCCCN(C(=O)C(O)Cc2ccccn2)C(C)C)cnn(C2CC2)c1 2243,c1(CC(=O)NCC2(C)CCC(NC(=O)C(N)=O)C2)ccc2c(c1)OC(F)(F)O2 2244,c1(NCCCC(=O)NCC2C(NC(C(C=C)O)=O)C2)ccc(C)cc1 2245,C(=O)(C(C)(C)C(=O)N1CC(CCCCNC(=O)CCC2CC2(Cl)Cl)C1)OC 2246,c1(C(=O)NC(C(C(C)C)NC(c2ccccc2O)=O)C)cncn(C)c1=O 2247,N1(C(C2CCCN(C)C2)=O)CCC(F)(CNC(c2sccc2C2CC2)=O)CC1 2248,CC1CCN(C(c2cccc(C3CC3)c2)=O)CCN1C(=O)Cc1ncc(Cl)s1 2249,C(=O)(CCCCCCS(N)(=O)=O)NC(CC)CNC(=O)Cc1cnn(CC)c1 2250,c1(CC(N2CCOCC(NC(c3ccn(C)c3)=O)C2)=O)cnc2ncccn12 2251,c1(C(N2C(C)CC(NC(C=C(C)C)=O)C2)=O)[nH]c2c(c1C)CCCC2 2252,C1(CC)CCCCCCN1C(=O)CC(C)CNC(C1(CF)CC1)=O 2253,C(=O)(CC1=NNC(=O)C1)NC1C(C)CCN(C(c2cc(C(F)F)c(Cl)cn2)=O)C1 2254,CCS(=O)(=O)c1ccc(CCC(=O)NC(CNC(C2(O)COC2)=O)CO)cc1 2255,C=C=C(C)CC(=O)NCC(CNC(c1ccc(OC(C)C)nn1)=O)CO 2256,N1(Cc2nnc(C(C)C)o2)CCC(NC(c2c[nH]c(Br)c2)=O)C(C)C1 2257,C(CO)(C=O)NCC(C)(C)NCCC(C)C.C(C)(C)(C)OC(C)=O 2258,c1(NC(C2N(C(c3cc(C)no3)=O)CC(F)C2)=O)cc2nccn2cn1 2259,Cc1nn(CC(C)C)c(C)c1CNC(C12CCC(CN1C(=O)OC(C)(C)C)C2)C 2260,CCC(C)C(C(=O)NC1CC(SC)C1)N(C)C(C1CC2CC1CC2O)=O 2261,CCC(CC)CCC(=O)NC1(C(=O)NC2CCOC(C)(C)C2)CC1 2262,c1(NC(c2ccc(CNC(CCC(C)OC)=O)cn2)=O)ccc2c(c1)OCC2 2263,N1(C(CS(CC)=O)=O)CCN(C(c2cn(C3CC3)nc2C)=O)C2(CC2)C1 2264,N1(C(c2n(C=C)nnc2)=O)CCOC2(CCN(C(=O)CC(C)(O)COC)C2)C1 2265,c1(C(N(C)CC2C3CN(C(CCC(=C)Cl)=O)CC32)=O)cc(C)c(=O)n(C)c1 2266,C(CCC(N)=O)(C(=O)NCC1CCN(C(c2cc(O)n(C)n2)=O)CC1)NC(C)=O 2267,C(=O)(C(C)(C)CC#N)NCCCC(C)(C)c1cn(CCC(CC)O)nn1 2268,c1(COC(C2(O)CCOCC2)=O)ccnc(CNc2ccc(OC(F)F)cn2)c1 2269,N1(C(C(C(C)O)NC(C)=O)=O)CCc2ccccc2C(NC(=O)C(C)C(C)C)C1 2270,N1(C(c2c(C)nc(C)s2)=O)CCN(C(c2cccc(Cl)c2O)=O)C(C2CC2)C1 2271,Cc1ccc(C(N2CCN(C(=O)C(N3CCCC3)C3CC3)CC2C)=O)c(C)n1 2272,C12(C(=O)NCC3CN(C(CC4CC(=C)C4)=O)CC3(C)C)CC1COC21CCC1 2273,O=C1CCC(C(N2CCN(C3CN(C(=O)C(Cl)=CCl)C3)CC2)=O)CN1 2274,Cc1cc[nH]c(=N)c1C(=O)NCC(C)NC(c1cnn(-c2cccc(F)c2)c1)=O 2275,C(CC(C(=O)N1CSCC1C(N1CCC(CCCO)CC1)=O)OC)OC 2276,c1(C(=O)OCc2n(C)cc(C(=O)OC)n2)cc(C)cc2c1CCC2 2277,N1(C(CCc2ccn(C)n2)=O)CC(CNC(C2(C#N)CC3CC3C2)=O)C(C)(C)C1 2278,C(=O)(C(CC(C)C)C(C)C)N(CC(C)NC(c1c(C)cc(C)nc1S)=O)C 2279,c1(C(=O)NCCN(C(=O)CC2CC2(C)C)C)cccnn1 2280,N1(C(c2c(C)nn[nH]2)=O)CCN(C(=O)Cc2nc(C3CC3)n[nH]2)C(CCO)C1 2281,C(=O)(CC(CC)C(C)C)N1CCCC(CN(C(=O)C(n2cc(C)cn2)C)CC)C1 2282,C1(NC(C2(C)CC(=C)C2)=O)CN(C(c2cnn(C(C)C)c2C)=O)CC1C(F)F 2283,c1(C(=O)NC2C(CNC(CCCc3onc(C)n3)=O)CCC2)cc(F)ccc1N 2284,c1(C(=O)NCC2N(C(C3CCN(CC)C3)=O)CCOC2)[nH]cc2c1CCCC2 2285,N1(C(c2nccc(C)c2)=O)CCC2CCC(C1)N2C(C1CN=C2N=CNN2C1)=O 2286,C(C(C)CN=c1cc[nH]c(C(=O)OC(C)=O)n1)NC(C(COC)(F)F)=O 2287,c1(C(=O)NCc2occ(C(=O)NC(CCC)(C)C)n2)cccc(O)c1C 2288,C=C=CC(C)C(=O)NC1CC(C)(NC(=O)CSc2ccc(C(C)(C)C)cc2)C1 2289,N1(C(c2c(O)ccc(CC)c2)=O)CCC2(CCN(C(=O)C(F)=CCCF)C2)C1 2290,c1(CCC(=O)NC2CCCC(NC(=O)Cn3ccnn3)C2)cccc(F)c1Cl 2291,C(=O)(CCC(=O)N1CCCC1(CC(C)C)C(=O)O)OCC 2292,n1(CC)ncc(C(N2CCCC(CNC(c3cc(F)n(C)n3)=O)C2)=O)c1C1CC1 2293,FC1(F)C2(NCc3nccn3-c3ccc(F)cc3)CCCCC12 2294,C1(NC(c2cc(OCC)ncc2)=O)C2CC1CN(C(c1cscn1)=O)C2 2295,CC(CC(=O)N1C2CCC1(CNC(=O)CC1CC1(C)C)CC2)C(F)(F)F 2296,C1(CNC(CC2(OC)CCC2)=O)CCC(NC(=O)COCc2ncc(C)o2)C1 2297,c1(CNC(C(C)OCCOC)=O)cccc(CN(C)C(c2sc(C)nc2C)=O)c1 2298,N1(C(C(CCC)OC)=O)CC2(CCCCN(C(=O)C(c3cncc(F)c3)C)C2)C1 2299,c1(CN(C)CC2CCCN(C(C3C(CC)CCCC3)=O)C2)ccc(O)c(O)c1 2300,C1(C(=O)NC(CCC)C)CN(C(=O)CCCF)CCC1(C)C 2301,c1(C(=O)NCCN(C(=O)Cn2cccnc2=O)CC)c(C)ncn1O 2302,c1(NCC2(O)CCN(C(CCC#C)=O)C2)cc(C)ccc1-n1ccnc1.C1(NC)CC1 2303,c1(C(=O)NCC2(CNC(c3cc(COC)no3)=O)CC2(F)F)cnc[nH]c1=N 2304,c1(C(=O)NCCCC2N(C(C(C)SC(C)C)=O)CCC2)cc(Br)n(C)c1 2305,c1(C(N(C)CC2N(C(c3cc(C)nnc3)=O)CCOC2)=O)c(C)nn(C)c1C 2306,C1(NC(=O)Cn2cnnn2)CN(C(c2cc(F)c[nH]2)=O)CC2(CCC2)C1 2307,c1(CC)[nH]ccc1C(=O)N(CCCCNC(c1ccsc1COC)=O)C 2308,c1(NC(c2cc(CCNC(C(CC)O)=O)on2)=O)ccc(N=[N+]=[N-])cc1 2309,C(=O)(C(C)(C)CC(=O)N(C)CC1(O)CCN(C(=O)C2=NNC(=O)CC2)CC1)OC 2310,C(Cc1ccccc1)(CCNC(=O)CN(C1CCC1)C)NC(C(C)O)=O 2311,N1(C(c2csc(Cl)c2)=O)CCCN(C(=O)C(O)C2CCCC2)C(CO)C1 2312,O=C(C1NCCc2ccccc21)NCC(C1CCCCC1)=O 2313,c1(C(=O)NC(C2OCCN(C(C(C)=CC3CC3)=O)C2)C)cncc([N+](=O)[O-])c1 2314,CCC(F)(CNC(=O)NC(C1CS(=O)(=O)C1)C)CC 2315,c1(CNC(C=C(C)C(F)F)=O)nc(CNC(=O)CCc2nccn2C)cs1 2316,c1(C(=O)NCC2CCCC(NC(C(C#C)(C)C)=O)C2)nccc(F)c1Cl 2317,c1(C(=O)NCC(CNC(C2(OC)CCOC2)=O)OC)cc(C2CC2)n(C)n1 2318,C1(CN(C)C(C2(NC(=O)CC3CS(=O)(=O)C3)CC2(C)C)=O)COC(=O)N1 2319,C1(NC(c2c(C)nn[nH]2)=O)CCN(C(=O)Cc2cc(F)cc(Cl)c2)C(C2CC2)C1 2320,C12(C(=O)NCCCC(C)NC(c3ccc(C4CC4)cn3)=O)CCC(CC1)CO2 2321,c1(C(=O)NCC(C)CNC(c2cc[nH]c2)=O)cc(OC(F)(F)F)ccc1F 2322,n1(-c2ccc(N(C(=O)CC(CC=C)OC)CC#C)cc2)ccc2cccnc12 2323,C1(C(C(=O)NC(C(C)C)CN2CCOCC2)Cc2ccccc2)CCCC(=O)N1 2324,CC1CN(C)CCC1N=c1nc2scnc2c(N2CCc3cc(F)ccc3C2)[nH]1 2325,C1(NC(C2(C)CC(=O)C23CCC3)=O)COc2cc(C(=O)O)nn2C1 2326,c1(C(=O)NCC23CCC(CN(C(CNC(C)=O)=O)C2)C3)ccc2[nH]c(=N)[nH]c2c1 2327,Cc1cc(C(=O)NCCN(C(=O)C(C)n2ccnn2)C)c2c(C)nn(C)c2n1 2328,C(C(O)CC(=O)NC(C)(C)CN(C)C)NC(COCCC(C)C)=O 2329,c1(NC23C(CN(C(C(CC)C(C)C)=O)C2)CCC3)ncc([N+](=O)[O-])cc1C(N)=O 2330,CC1=CCC(C(=O)NCC23CC(NC(c4cnn(C(C)(C)C)c4N)=O)(C2)C3)CC1 2331,C1(CC(=O)NCC2(F)CN(C(c3ccc(C(F)(F)F)cc3)=O)C2)CCCC1(F)F 2332,N1(C(Cc2c(C)nc[nH]2)=O)CCC(NC(=O)CCc2cncn2C)C12CCC2 2333,CCC(CCC(=O)NCCOCC1CCCC1)NC(=O)CS(=O)CC 2334,c1(NC(=O)NNC(=O)c2ccccc2F)ccc2cc[nH]c2n1 2335,c1(NC(C2C(NC(CCCOC)=O)CC2)=O)ccc(SC)nc1 2336,C1(CC(C)C)CCN(CCCc2nnc(-c3cccs3)o2)CC1 2337,C1(NC(C(Cn2cncn2)NC(c2ncc(OC)nc2)=O)=O)CCOCC1(C)C 2338,CC1(C)C(C(=O)NCC(CO)NC(=O)C2=NOCC2)CC1(F)F 2339,N1(C(CC2(OCC)CCC2)=O)CCC2(CC2)CC1C(N1CC2CC2C2CC12)=O 2340,Cc1noc(Cl)c1CC(N1CCCC(c2cn(CCN(C)C)nn2)C1)=O 2341,N1(C(CCC)=O)CC2CC1CN2C(=O)Cc1cc(Cl)ccc1Br 2342,c1(CC(CC)C)nc(-c2nn(C)nc2Br)n(-c2cnnn2C)n1 2343,Cc1ccc(C(N2CCC2C(N2CC(CC(N)=O)C2)=O)=O)[nH]1 2344,Cc1ccn(CC(=O)N(CCNC(=O)Cc2nc[nH]n2)C(C)C)n1 2345,C=CCC(C)C(=O)NC1CC(NC(=O)CCSc2nccn2C)C1 2346,c1(OC)cc(C(N2CC(CC(C)NC(c3csc(Cl)n3)=O)C2)=O)cc(F)c1 2347,c1(C(=O)NCC(CC)NC(C2CCCC23CC3)=O)cnn(C(C)(C)C)c1Cl 2348,Cc1nn(CC(=O)NCC#CCNC(C2CC23CCCC3)=O)c(C)c1C=NO 2349,CC(C)(C(=O)NC1CC(F)CN(C(c2cc(C3CCOCC3)[nH]n2)=O)C1)C(N)=O 2350,C1(C(N2CCN(C)CC2CNC(=O)Cn2cnnc2)=O)CCCC2CCCCC12 2351,C(=O)(CCC1=CCCCC1)N(CCC(C)NC(=O)CC(C)O)C 2352,N1(C(C)C)CC(NC(=NCc2ccccc2)NCc2nncn2C2CC2)CCC1=O 2353,S(=O)(=O)(c1ccc(NCC(C)C)cc1Br)NC(C)CN1CCOCC1.C(CCC#N)S 2354,CON(CCC(=O)NC(C)C(F)F)C(=O)C1CC(C(C)C)C1 2355,c1(C(=O)NC2CC(C)(c3nc(CCC(O)CCO)no3)C2)cc2ncccn2n1 2356,N1(C(c2cc(C)cc(C)c2)=O)CCN(C(c2nnsc2C)=O)C2CCCCC12 2357,CC1CC(NC(c2cc(Cl)c(Cl)s2)=O)CN(C(=O)Cc2cc(F)ccc2O)C1 2358,C12(C(=O)NCCCCNC(C(CC)OC)=O)CC(c3ccccc3)(C1)C2(F)F 2359,C1(NC(=O)NCCC(C)SC)CC(=NOCC#N)C1 2360,C1(C(C)(C)NC(=O)Cn2ncnn2)CCCCN1C(=O)CC1(O)CCC1 2361,C=CC(C)(O)C(=O)N(C1CCN(C(=O)C(C)=CCN(C)C)CC1)CCOC(C)=O 2362,C1(CCOC)CN(C(=O)CC(C)COC)CCN1C(=O)C(C)Cc1cnc[nH]1 2363,c1(C(=O)NC2(CNC(c3ccnnc3S)=O)CCOC2)ccc(Cl)cc1Cl 2364,Cc1cc(P(C)(C)=O)oc1C(N1CCN(C(=O)Cn2cc([N+](=O)[O-])cn2)CC1)=O 2365,N1(C(C2CCC(CNC(C3(C4(C)CC4)CC3)=O)CC2)=O)Cc2cncnc2C1 2366,C(=O)(C(C)(CO)NC(=O)C(c1cnn(C)c1)C)NC(CC(C)C)C 2367,c1(CNC(CCN(C)C(C2CCCN2C)=O)=O)ncc(Cl)cn1 2368,c1(C(=O)NC2C(C)N(C(c3csc(C(F)F)n3)=O)CC2)cccc2nn(C)cc12 2369,c1(NC(C(C=C)F)=O)ccccc1NC(=O)CCc1ccc(C)cc1 2370,C(C)(CO)(C(=O)N(C)CC1(CNC(=O)CCn2ccnc2C)CC1)NC(C)=O 2371,N1(C(C2C(COC)CC2)=O)CC2CN(C(=O)CN3CCCS3(=O)=O)CC2(C)C1 2372,CC1CCN(C(c2cccc3c2CCC3)=O)CCN1C(c1ccn2c1CCC2)=O 2373,CC1=C(C(=O)N2CCCC2CCCCNC(c2cnc(O)c(Br)c2)=O)CCO1 2374,C1(C(=O)NC(C(=O)NC(C(=O)N(CC)CC)C)c2ccoc2)CCC=CCCC1 2375,Cc1ccccc1CN(C(=O)C(c1ccoc1)NC(=O)COC1CC1)C 2376,C=C(C)C1CN(C(=O)CCCC(C)NC(=O)C(C)CC=O)CCO1 2377,c1(C(N2C3(CNC(c4cc(C)[nH]n4)=O)CCC3CC2)=O)cc(S(C)(=O)=O)cs1 2378,N1(C(C(C)=CC)=O)CCC(NC(c2nccc(OC)c2OC)=O)C(CC)C1 2379,Cc1cccc(N)c1C(N1CC(CCNC(c2ccnn2C(C)C)=O)C(C)C1)=O 2380,CC1(S(C)(=O)=O)CCCC1C(=O)NCC1CCN(C(=O)CSCC(N)=O)C12CC2 2381,CCC(C)C(C)C(=O)NCCCCn1cc(-c2cn(C)nc2C(=O)OC)nn1 2382,c1(CNC)ccc(NC(c2sc(C(C)C)nc2C)=O)cc1 2383,CC1CN(C(=O)Cc2ccn(C)n2)CC1(C)CNC(=O)Cn1ccccc1=O 2384,c1(C(=O)OC)cn(C)nc1C(=O)NC(C)CN(C(=O)CC12CCCC1C2)C 2385,Cc1cc(C)c(C(=O)NCC2C=CCN2C(=O)CN2CCCCCC2)s1 2386,Cc1cc(C(=O)N(CCCN(C)C(c2cc(=O)n(C)cn2)=O)C)nc(O)c1 2387,c1(N2CCC(C(C)C)C2)nc(N2CCC(C)(c3ccccc3)C2)c2ncsc2n1 2388,C=C(C)CC(C(=O)N1CCC1CNC(=O)CSc1csc(C)n1)NC(C)=O 2389,CS(=O)(=O)c1cc(C(=O)NCCc2ccn(CC(F)(F)F)n2)c(Cl)cn1 2390,CS(=O)(=O)C1(C(=O)NCC2CC3CN(C(=O)C4=COCC4)CC23)CCCC1 2391,N1(C(C(Br)=C(C)C)=O)CCC(C2CC2)(CNC(c2ncnc3c2CCC3)=O)C1 2392,C1(C(N2CCSCC(C)C2)=O)COC2(C1)CN(C(c1c[nH]c(C#N)c1)=O)C2 2393,N1(C(c2cc(C)c(Cl)s2)=O)CCN(C(=O)Cc2conc2C)C2CC12 2394,N1(C(C2C(C)OCC2)=O)CCC2OCCN(C(c3ns[nH]c3=O)=O)C2C1 2395,c1(C(N(C)CC2C3CN(C(C(CCC)C#N)=O)CC32)=O)cc(Cl)c(F)cc1OC 2396,c1(C(=O)OC)c[nH]ccc1=NCC1(O)CCCN(C(=O)C=Cc2cn(C)nn2)C1 2397,C1(OCC)CC2CN(C(=O)C(CN(C)C)NC(c3c(C)noc3N)=O)CC12 2398,c1(N2CC(C=C)OCC2)cc(S(=O)(=O)NC2CC3(CC3)C2)ccc1C#N 2399,c1(C(N2C3CN(C(C(C)O)=O)C(C3)C2)=O)ccc2c(O)nnc(O)c2c1 2400,c1(C(=O)NC2CN(C(c3c(CC)n(C)cc3)=O)C3C2C3)ccc([N+](=O)[O-])cn1 2401,C1(CC(=O)NCC(CC)N(C)C(c2n[nH]c(C)c2C)=O)OCCCC1(C)C 2402,Cc1cc(Cl)cc(C)c1C(=O)NC1CC(NC(=O)CC(C)(C(F)F)N(C)C)C1 2403,C12(CNC(c3n(CC#C)ccc3)=O)CN(C(=O)CN3CCCC3)C(COC)(C1)C2 2404,C1(N(C(CCC(C)OC)=O)C)CN(C(=O)CSc2ccc(F)cc2F)CC12CC2 2405,C1(C(N(C)Cc2ccn(CC)n2)=O)CN(C(=O)C(C)OCCOC)C(C)(C)C1 2406,N1(C(CNC(CN(S(C)(=O)=O)C)=O)C(F)F)CCN(C(C2(C)CC(C)C2)=O)CC1 2407,C(C(C)C(F)C(=O)N(CCCN(C)C)C)NC(C1(OCC)CC1)=O 2408,C1(C(=O)NC2CC(CNC(COCC=C)=O)C2)CC2(C1)CC1(CCC1)C2 2409,C1(CN(C)C(C2CC(C)(NC(=O)C(C3CC3)C3CC3)C2)=O)CCCCO1 2410,C1(CC)C(NC(c2cnc(CC(C)(C)C)o2)=O)CCCN1C(c1cnco1)=O 2411,c1(C(N2C(CNC(C3N(N=O)CCCC3)=O)C=CC2)=O)ncnc2ccsc12 2412,N1(C(C2N(CCC)CCC2)=O)C(C)CN(C(C2(C)CC=CC2)=O)CC1C 2413,CC(C)(C)CC(O)C(=O)N1CCN(C(=O)CNC(N)=O)CC(CO)C1 2414,Cn1ncc2ncnc(N3CCN(C(=O)CCc4nccs4)CC3CCO)c12 2415,C(C(C)(C)CNC(C1CCCN1c1nccs1)=O)N(C(=O)C=CC(F)(F)F)C 2416,Cn1c(O)nc2c(C(=O)NC3CCN(C(c4cnc(O)s4)=O)CC3F)cccc12 2417,c1(SC)cc(C(=O)NCC(C2CCN(C(=O)C(O)c3ccco3)CC2)C)oc1C 2418,c1(C(N(CC(C)CNC(c2cccnc2Cl)=O)C)=O)ccnc2c1CC(=O)N2 2419,n1(CC(=O)NC2CC(CNC(C(c3ccccc3)OC)=O)C2)nnnc1C1CC1 2420,N1(C(C(C(=C)C)(C)C)=O)CC(NC(=O)C(C)(C2CC2)OC)CC2(CCC2)C1 2421,c1(C(N2CCN(C(c3ccnc(C)c3N)=O)CC2CO)=O)ccc(S(C)(=O)=O)o1 2422,C(=O)(C#CC1(C)CCCO1)NC(CC(C)NC(c1nnc(C(C)C)s1)=O)C 2423,C1(N(C(=O)CC2CC2)CC2CCOCC2)CCCCC1 2424,C1(C(N2CC(C(C)NC(C3CCC(=O)O3)=O)C2)=O)CCC2CC2CC1 2425,O=S(=O)(c1ccc(NCc2cscn2)c(F)c1)N1CC2CC3CC2C1C3O 2426,C1(CN(C(c2cc(CNC(c3scc(C)c3)=O)oc2)=O)C2CC2)CCCC(C)C1 2427,N1(C(Cn2nc(C)n(C)c2=O)=O)CCC2CCN(C(C3(C)CC3(F)Cl)=O)CC2C1 2428,C1(C(=O)NCC(CCNC(CNC=O)=O)O)CCCN1N=O 2429,CCC(C(=O)NCC(Cc1ccccc1)N(C)C(C12CC(CO1)C2)=O)N(C)C 2430,C(=O)(C(F)C1=CCCCC1)NC(CCNC(c1ncc(CC)s1)=O)C 2431,Cn1cnc(CCC(=O)NCCSCC(N2CC(OCC(N)=O)C2)=O)c1 2432,Cn1ncc(NC(C2(CCCF)CC2)=O)c1-n1cc(C2(N(C)C)CCOC2)nn1 2433,C1(C)(C(=O)OC)CCN(C(C2CCN(C(C3CC4CC4C3)=O)CC2)=O)C1 2434,C(=O)(CC1=NNC(=O)C1)N1CCC(NC(C(C)N(CC)CC)=O)C(C)C1 2435,C1(NC(CN(C(C)C)C(C2CCC3CC2CO3)=O)=O)CN2CCC1CC2 2436,n1(CC(=O)NC2CCN(C(=O)C=CC3CCCCC3)C2)nc(Cl)ccc1=O 2437,CCC(C(=O)N1CCCC(c2cn(C(C)(C)C(=O)OCC)nn2)C1)C(C)(C)CC 2438,C(=O)(C1CNC(=O)c2ccccc21)N1CC2C(NC(CCOC)=O)C(C2)C1 2439,C1(C(C(N2CC(CC=CC)C2)=O)C)CCCN(C(=O)C(C)=C(C)CC)C1 2440,CC(CCCCNC(c1cscc1Cl)=O)NC(=O)C(F)=C1CCCC1 2441,C1(CCCNC(C=C(C)C)=O)CCCCN1C(C12CC(C(C)C)(CO1)C2)=O 2442,C1(NC(CC(C)OC)=O)COC2(CNC(C3(CC4CC4)CCC3)=O)CC1C2 2443,c1(C(C)=O)ccccc1C(=O)NC1CCN(C(C)=O)C1C(=O)O 2444,c1(C(N2C(C(=O)NC3(CC#C)CC3)CC2C)=O)ccc(C)c(F)c1 2445,C1(C(F)(F)F)(C(N(C)CC2CN(C(CC3C(C)CCC3)=O)C2)=O)CCCCO1 2446,c1(NC(N2C(C(=O)Nc3ncn(CC)n3)CC2)=O)cc(OC)c(F)cc1F 2447,c1(C(=O)NCCCCCCNC(C2CC(CF)C2)=O)cccc2occc12 2448,C1(C2CCN(C(=O)CC3(C#N)CCC3)C2)(NC(COC(C)(C)C(F)(F)F)=O)CC1 2449,N1(C(C2=CC(C)(C)C2)=O)CC2CCN(C(=O)C3Cc4ccccc43)C(C2)C1 2450,Cc1oc(C(C)C)cc1C(=O)NCCC(O)CNC(C1CC1c1ccccc1)=O 2451,C(CCC(=O)NCC=CCNC(c1c[nH]cc1C(C)C)=O)=C(C)C 2452,C12(C(=O)NCC3C(CNC(C4C(c5n(C)ncc5)C4)=O)C3)CC1COC21CCC1 2453,C(=O)(CC(O)CC(C)(C)C)N1CC(NC(CCCOC)=O)C2(C1)CC2 2454,c1(NC)c(C(N2CCCC(NC(C3(C)CCC(F)(F)C3)=O)C2C)=O)cccc1N 2455,C12(C(N3CCC(NC(C4C(CC)C4)=O)(CC)CC3)=O)CCC(F)(CC1)CC2 2456,Cc1nscc1C(=O)NCCCC1CCCN1C(=O)COCC1CCCCO1 2457,N1(C(CCCC2C(C)C2)=O)CCOC(C(=O)NC(C(F)(F)F)C2CC2)CC1 2458,C1(CN(CC(=O)N(C2CCCCC2)CCC)C)CCN(C)C1 2459,N1(C(C2N(CC)CCCC2)=O)CCCC(C2CCN(C(=O)C(C)CCO)C2)C1 2460,c1(C(N2CCC(NC(CC=C(C)C)=O)C2C)=O)ccc2c(c1)CCC(C)(C)O2 2461,C1(C(N2CCC(O)(CN(C)C(C3C=CCC3)=O)CC2)=O)C2CCC1(C)C2(C)C 2462,N1(C(C(C)(C)SC)=O)CCC(C(C)(C)NC(=O)C(=O)NCC(F)(F)F)CC1 2463,c1(CC(=O)OC)ccccc1C(=O)NCC#CCNC(=O)CC1OCCC1(C)C 2464,S(=O)(=O)(c1ccc(F)cc1)NCCC(N1CCC(n2nnnc2C2CC2)CC1)=O 2465,c1(CCC(=O)Nc2cccc(C(=O)OCC)c2)ccc2ccn(C)c2c1 2466,C(CCC(=O)NCCC(=C)CNC(=O)C(C)NC(=O)CC1C=CCC1)=CCC=C 2467,C=C(Cl)CC(C(=O)N(C1CCCC1C)C)NC(C1CNC(=O)O1)=O 2468,c1(N(C(C)C)C)ncc(CN2CCSCC(C)C2)cc1F 2469,C1(N(C(C(CC)C)=O)C)CN(C(=O)Cn2nc(Cl)ccc2=O)CC1(C)C 2470,C(CN=C(NCc1ccccc1Cl)NCC1CCCCC1)C1CC(C)OCC1 2471,C12(C(=O)NCC=CCNC(c3cccc(O)c3F)=O)CCC(CC1)CC2 2472,C1(C(N2C(CNC(c3cc(C)sn3)=O)CCCC2)=O)CN2CCN1CC2C 2473,CCC(CC(F)(F)F)C(=O)NC(C)(CNC(=O)Cc1cc(C(F)(F)F)n[nH]1)CC 2474,C1(CNC(CCCCNC(C=CC(=O)OCC)=O)=O)CCCCC(O)C1 2475,C1(C(=O)OCCn2ccc3ccccc23)CC2(CCC2)C12CCC2 2476,c1(N(CC(=O)N(C)C)C)ccc(S(=O)(=O)NCCC(CO)C2CCC2)c(Br)c1 2477,N1(C(CNC(C2(C#N)CC2)=O)=O)CCN(C(=O)CC2CC3(CC3)CO2)CC1 2478,c1(C(=O)NCCCCC(C)NC(=O)CSCC(N)=O)cccc(C#N)c1Br 2479,C1(NC(c2c(C3C(C)C3)noc2)=O)CC(F)CN(C(=O)Cc2cn(C)nn2)C1 2480,c1(C(=O)NCCCCN(C(=O)Cn2cnnn2)C)sccc1Cl 2481,CC1CN(C(=O)CC2CCN(C(c3ccn4c3CCC4)=O)C2)CC(=O)N1C 2482,N1(C(CCCOCCOCC#C)=O)CC(NC(=O)COC(C)=O)C2(CC2)C1 2483,c1(CCC)c(C(N2CC(CNC(c3occc3C)=O)CC2C)=O)nnn1CC 2484,N1(C(CC(C)=C(C)C)=O)CCC(C)(CCNC(c2ccc(C3CC3)o2)=O)C1 2485,c1(C(N2CCOC(CCCNC(=O)C3CC3)C2)C(=O)NC)ccc(C2CC2)cc1 2486,c1(CN2C(CC(=O)Nc3ccc(C(=O)NC)cn3)CCC2)cc(Cl)c(Cl)cc1C 2487,c1(CC)c(C(=O)NCCC(C)(C)NC(=O)CCc2ncc(F)cn2)csc1C 2488,N1(C(c2nc(CC)oc2C)=O)CCN(C(c2ns[nH]c2=O)=O)CC2CCCCC12 2489,C(=O)(C1=CCC2CCC1N2C(=O)C(C(=O)OC)OC)N(CC)CC1CCOC1 2490,C1(O)(CCNC(c2cc(C)oc2)=O)CCN(C(C2CC(N(C)C)C2)=O)C1 2491,N1(C(C(c2ccc(Cl)s2)C)=O)CC=C(CNC(=O)C(F)C2CCC2)CC1 2492,N(C(=NCCN1CCC(C)C1)NC1CCN(C(=O)OC)CC1)CC(=C)C 2493,C(=O)(C1=NNC(=O)CC1)N1CCC(O)(C(=O)Nc2cc(OC)cc(Cl)n2)C1 2494,c1(CC(=O)N(C)CCOCCCNC(c2cnc[nH]2)=O)ccccc1Br 2495,C1(NC(C2CCCC23CC3)=O)COCCN(C(c2ccc(F)cc2F)=O)C1 2496,c1(C(C2(C(C)CNC(C3CC(CC)(CC)C3)=O)CC2)=O)cnn(C)c1C(C)C 2497,Cc1cnc(NC(C2CC23CN(C(c2cnc(Cl)cn2)=O)C3)=O)cc1F 2498,c1(C(C(=O)OC)N(C(=O)CC2CS(=O)(=O)C2)C)cccc(Cl)c1Cl 2499,C1(C(=O)OC)CC(n2cc(C3(C(C)=O)CC3)nn2)CN1C(c1cccc(C)c1)=O 2500,c1(CC)nn(C)c(Cc2nc(-c3ccn(C)n3)nn2CC2CC2C)c1Cl 2501,Cc1cccc2c1N(C(C1CCCC1NC(=O)CCC1CCCCO1)=O)CC2 2502,c1(C(=O)NCC2(CN=c3nc(C4CCCC4)[nH]s3)CCC2)cnc2[nH]cncc1-2 2503,c1(C(=O)NCC(CC)(C)NC(C2CCN(C)C2=O)=O)nccc2c1CNC2=O 2504,C1(C(=O)NC2C(=O)OCC2CO)(NC(C(C(C)C)F)=O)CCc2cc(Br)ccc2C1 2505,O=C1COc2ccc(C(=O)NC3CN(C(=O)C=CCF)CCC3F)cc2N1 2506,C(=O)(C(F)(F)Cc1ccccc1)N(C)CCNC(C12CC(CO1)C2)=O 2507,CCCCC(CCCC)NC(=O)CC(C)(C)N(C(=O)Cc1cccc(C#N)c1)C 2508,N1(C(C(CC)C)=O)Cc2ccccc2OC2(C1)CN(C(=O)Cc1ccc(C)o1)C2 2509,C(=O)(C1=NNC(C(F)(F)F)C1)NC1(CN(C(CN(C)CC)=O)CC)CCCC1 2510,c1(C(=O)NC(CC)CNC(=O)C(C)=C(C)C)ccc2nnnn2c1 2511,c1(OC)ncc(C(=O)NCC2(C)CN(C(=O)C(C)N(C)C)CCO2)nc1C 2512,N1(C(CCC2C(C)(C)C2)=O)CC2CC1(C(=O)NC1CCC(O)CC1)C2 2513,CC1CN2CCN1C(C(N1CCCCC1CNC(C1(C)COC(=O)C1)=O)=O)C2 2514,C1(C(N(CCCCCCNC(CCCC)=O)C)=O)C2CCC(C2)S1(=O)=O 2515,C(CC(=O)NCC1(NC(C2CC2CC)=O)CC1)OCC#C 2516,Cc1coc(C(N2CCC(N3CCC(NC(=O)C(=O)NC(C)C)CC3)C2)=O)c1C 2517,Cc1c(Cl)ccnc1C(=O)NCC1CC(F)CN1C(=O)CO 2518,CCC(CC(=O)N(C)CC1CN(C(c2n[nH]c(C3CC3)c2C)=O)CCO1)C(C)C 2519,N1(C2CN(C(=O)C(COC)NC(c3c[nH]nc3C(C)C)=O)C2)CC(CC)CC1=O 2520,C#CC1CN(C(=O)CCC2CCCN(C(=O)C(C)=C(C)CC)C2)CC1OC 2521,C#Cc1ccc(C(=O)NCCN(C(=O)Cc2conc2C)CC2CC2)cc1Cl 2522,N1(C(C2C(CNC(C3(CC#C)CCOC3)=O)OCC2)=O)CC2CSCC(C2)C1 2523,CC(CC(C)(C)C)C(=O)N(C1CCN(C(C2CCN(C)C(C)C2)=O)C1)CC1CC1 2524,CCC(CCOC)C(=O)NCC1(F)CN(C(C2Cc3nccn3C2)=O)C1 2525,c1(NC(C2CC(NC(CCCNC(C)=O)=O)C2)=O)ccc(Br)nc1 2526,C(c1cc(C)no1)=CCN(C(C(=O)NCCNS(CC)(=O)=O)C1CC1)C 2527,N1(C(C2N(C(CC(C(C)C)O)=O)CCSC2)=O)CC2(CCOC2=O)C1 2528,C1(C(=O)NCC(C)CNC(C2(C)CC(C#N)C2)=O)CC(c2cccc(F)c2)=NO1 2529,c1(C(N2CC(N(C(C(C=C)O)=O)C)C(O)C2)=O)nn(C)cc1S(N)(=O)=O 2530,C(=O)(C(C(=O)NC1(CNC(C2(C)CC(C)=NO2)=O)CCCCC1)C1CC1)OCC 2531,C1(OC)(CNC(c2cc(CO)ccn2)=O)CCN(C(=O)C(C)(F)F)C1 2532,C1(CNC(C2(CC#C)CCC2)=O)CN(C(c2cnc(C(C)OC)[nH]2)=O)CC1(F)F 2533,CCCC(C)C(=O)N1CCC(C2OCCCC2NC(=O)CCc2cnco2)CC1 2534,C12(NC(C=COCC)=O)CCCC1N(C(c1cncs1)=O)CC2 2535,c1(SCC)cnc(O)c(C(N2CC(NC(C3(C(C)C)CC3)=O)C(C)C2)=O)c1 2536,N1(C(C(C)C2CC2)=O)CCN(C(C2CCC(OC(F)F)CC2)=O)CC1C 2537,N1(C(C)C)CCCC1CC(=O)N(C(C)CCNC(=O)CCCN(C)C)C 2538,C(N=c1cc[nH]c(=NCCc2cccc(Cl)c2Cl)[nH]1)c1coc(C)c1C(N)=O 2539,C(CCN(C)C(C1(Cl)CC1(C)C)=O)(C(C)C)NC(c1cc(CCCCC)[nH]n1)=O 2540,N1(C(c2ccc(CC)s2)=O)CCC(C)C(NC(=O)CCC(F)F)C1C 2541,CC1(C2CCCN(C(=O)CC3CCCN(C(c4cn[nH]c4)=O)C3)C2)CC1 2542,N1(C(CN(C2C=CS(=O)(=O)C2)CC)=O)CCCC2(C1)NC(=O)N(C)C2=O 2543,C1(C(C)C)C(NC(C2CC3(CCC3)C2)=O)CCN1C(=O)COC1(C)CCCC1 2544,c1(CN2C(CCCNC(C3N(C(=O)NC)CCC3)=O)CCC2)cccc(C)c1 2545,C1(NC(C(CC#CC)NC(c2cc(CCC)[nH]n2)=O)=O)CCN(C)CC1C#N 2546,N1(C(C2(CC=C)CCOC2)=O)CC(C2CCCN(C(=O)CN(C)C)C2)C1 2547,C1(CC)CCC(C)CN1C(C1CN(C(c2cocc2C(N)=O)=O)CCN1C)=O 2548,C12CCCCN1C2.c1(SCCCN2CC(O)C2)nnnn1-c1cccs1 2549,c1(CC(=O)N(CCCNC(c2cccn2C)=O)C(C)C)cccc2ccccc12 2550,C(=O)(CC(C(F)F)n1ccnc1)NC(CN(C)Cc1nc(C(C)C)sc1)C 2551,C(=O)(N=c1[nH][nH]c2c1CNC2(C)C)C1CC1.c1(NS(CC)(=O)=O)ccc2ncsc2c1 2552,c1(C(=O)NC(C(C(=O)N(CC(=C)C)C)C)C)ccc(=NC)[nH]c1 2553,C(=O)(CC(F)(F)C(C)C)N1CC(CCNC(C2N(CC)CCCC2)=O)OCCC1 2554,c1(C(N2CCC(CN(C(C(CC)(C)OC)=O)C)CC2)=O)ncncc1C#N 2555,O=C(C(O)C(F)(F)F)NC1CCCS(=O)(=O)C1 2556,C=Cc1cncc(C(=O)NCC2CC3CC3N2C(c2cc(C3CCC3)[nH]n2)=O)c1 2557,CN1CCC(C(=O)NCC2N(C(c3cnn(CO)n3)=O)CCC2(C)C)CC1=O 2558,c1(CN2CCCC(NC(c3ccc(CN(C)C)cc3)=O)C2)ccc(F)c(C#N)c1 2559,C1(CSCC(=O)NCCCNC(Cc2nc(C)oc2)=O)CCc2ccccc2O1 2560,C(=O)(CC1OCc2ncccc21)NCCCN(C(C(CCSC)O)=O)C(C)C 2561,c1(CNC(c2ccc(CNC(C3N(C(C)(C)C)CC3)=O)s2)=O)csc(C#N)c1 2562,N1(C(C2(F)CCN(C(c3ccnc(F)c3Cl)=O)C2)=O)CCN2CCCC2C1 2563,C(C(C)C(=O)NCCC(Cc1ccccc1)NC(c1nscc1N)=O)SC 2564,CC(C)C(C)C(CNC(C1CCCCC1)=O)NC(c1cn(C)nc1C(C)(F)F)=O 2565,N1(C(c2scc(C)c2)=O)CCCCC2(CCN(CC(=O)NCc3cccs3)C2)C1 2566,CCC(C)CCCC(=O)N1CC2(CC2)CC1C(N1CCC2(CC1)N=N2)=O 2567,C(CCCC(C)NC(c1cnc(Cl)s1)=O)NC(C1(CC)CC1(F)F)=O 2568,C1(C(=O)NC(CSC)C)CC2CC1CN(C(c1ccc(O)cc1F)=O)C2 2569,C=C(C)C1OCCCC1C(=O)NCC1CCCN1C(c1cnn(C)c1SC)=O 2570,C(=O)(CC(O)C(C)C)NC(CCCNC(c1[nH]c(=NCC)sc1)=O)C 2571,C1(CC#C)(C(N2CC(CC=C)(NC(=O)C(O)Cc3cnc[nH]3)C2)=O)CCCCO1 2572,N1(C(C2(CC)CC2)=O)CCOC(C)(C)CC1 2573,C1(C(N2CCC(C)(F)C2)=O)N(C(=O)Cc2nc(=N)[nH][nH]2)CC12CCCC2 2574,c1(CC)n[nH]c(CC)c1CC(=O)NCC12CC1CN(C(C1(C)CC(F)C1)=O)C2 2575,C(=O)(C(C)(C)CC#N)NC(C(C)C)CCNC(=O)C(C)Sc1ccccc1 2576,C#Cc1cn(C)nc1C(=O)NCCCCN(C(=O)C(C)(C)C#C)C 2577,c1(N2CCC3(CC(OC)C3)C2)ncnc2[nH]cc(C(=O)O)c12 2578,C1(CNC(C2(C(CC)(F)F)CC2)=O)(NC(=O)Cc2ncccc2C)CCOCC1 2579,N1(C(C(CC)Sc2ccccc2)=O)CCC(O)(C2(NC(=O)C(C)O)CC2)CC1 2580,C1(CNC(C2(CC)CC2)=O)CN(C(=O)Cc2cn3ccccc3n2)CCC1(C)C 2581,c1(OC)c(C)n[nH]c1C.C(CCC(=O)N1CCC(C2CCCN2CC)C1)OCCO 2582,C(=O)(CC(C)C(C)C)NCC(CC(C)C)NC(c1scnc1C1CCCCC1)=O 2583,C1(CC(=O)NC2CCC(N(C)C(c3cc(CO)on3)=O)C2)CC2CCC1CC2 2584,CN1CCN(C(C2CCS2(=O)=O)=O)C(CNC(c2cccnc2O)=O)C1 2585,CC1(C)OC2(CNC(C3CC34CCCOC4)=O)CC1(NC(=O)C1=C(Cl)CC1)C2 2586,C1(CNC(CCc2cccc(OC)n2)=O)CCCCN(C(=O)CCS(C)(=O)=O)C1 2587,C(CC=C)(CC(=O)N(CC(C1CCCC1)O)C)NC(C(C=C=C)C)=O 2588,C(C(=O)O)(C(C)OC)CC1CCN(CCCOC)C1.C(C)(C)(C)OC 2589,Cc1c(C(=O)NC2CCC23CN(C(C2COC(=O)C2)=O)C3)oc2ccc(F)cc12 2590,Cc1c(NC(=O)CN2CCN(C(c3ccccc3O)=O)CC2)cnn1C 2591,C1(NC(C2(C)SCCCS2)=O)CCCC(C(=O)NOCCCC2CC2)CC1 2592,C1(C(=O)NC2(CC=C)CC2)CN(C(c2c(C)cccc2C)=O)CCC1(C)C 2593,c1(N(C(C)CCNC(c2ncn3ccccc23)=O)C)ncnc(Cl)c1C#N 2594,C=C(C)CCCC(=O)N1CC(NC(c2c[nH]cc(Cl)c2=O)=O)C(C)C1 2595,CCC1=C(C(=O)N(C(CNC(=O)Cn2ncc(O)nc2=O)C2CC2)C)CCCO1 2596,c1(C(N2C(C(=O)NC3CCSC3)(COC)C=CC2)=O)ccnc(O)c1F 2597,c1(C(=O)OC(Cc2ccc(OC)cc2)C)ccc2cc(OC)ccc2c1 2598,S(=O)(=O)(C1CN(C(=O)CCC(C)O)C1)N1CCN(C(CCSCCCC)=O)CC1 2599,N1(C(Cn2c(C)ccn2)=O)CCC2CCN(C(=O)CCC3CCCCO3)CC12 2600,c1(OCC)ccc(F)cc1CC(=O)NCC(C1CCC1)NC(c1ncsc1C)=O 2601,c1(N(CCCC)C)ccnc(C(N2CCC(NC(c3ccc(Cl)s3)=O)CC2)=O)n1 2602,C1(C)(NC(C(C)NC(c2cn(C(C)C)nc2)=O)=O)CN2CCC1CC2 2603,c1(CC(=O)NC(CC(=O)N2CC(C)C2)Cc2cccc(Br)c2)cc(Br)ccc1O 2604,C=CCC(C(=O)N1CC(CNC(=O)Cc2nocc2C)OC(C)(C)C1)C(C)C 2605,N1(C(CC(COC)C)=O)CCC(F)(CNC(C2(C)CCC(C)C2)=O)CC1 2606,C1(=CCC)CN(C(=O)C(C)NC(=O)C(C)SC)C1 2607,C1(NC(CC2(OC)CCCC2)=O)CCN(C(c2nocc2C(C)(C)C)=O)CC1C 2608,C1(CN(C(=O)CCn2ccccc2=O)C)CN(C(c2ccsc2)=O)CC12CC2 2609,Cn1ccc2c(C(=O)NC3CC(O)CN(C(c4coc(Cl)n4)=O)C3)[nH]cc2c1=O 2610,C1(CNC(CCCC=C)=O)(OC)CCN(C(c2ccnn2CCF)=O)CC1 2611,C1(Cn2cc(C(C)O)nn2)CN(C(c2csc(-c3ccoc3)n2)=O)CCO1 2612,N1(C(c2cc(CNC(C(CC)(C)CC)=O)on2)=O)CC(C)CC(C)(C)C1 2613,C12(CC1)C(=O)N2.C(CCN(C(=O)CN(C)CC)C(C)C)OCC 2614,N1(C(c2cccnc2)=O)CCC(O)(c2cccc(Cl)c2)CC1.O=C1CC2CN1C2 2615,c1(C(=O)NC(c2nocc2C(=O)NCC(F)F)C)sccc1C#N 2616,C1(C)(CC)C=C(C(=O)N2CC(CNC(=O)CCc3nccs3)C(O)C2)C1 2617,N1(C(c2nccc(C#C)c2)=O)CCC(C(=O)NCC(F)(F)CO)=C(F)C1 2618,C1(OCC)CCN(C(=O)C(C)(C)NC(C2CCC(F)C2)=O)CC1 2619,CC(=O)CCCCC(=O)NCC(C)(C)OCC(=O)NC(C1CC=CCC1)CO 2620,N1(C(c2ncn(C)n2)=O)CC(O)CC1CNC(c1cc(C2CC2)n(C)n1)=O 2621,C1(CNC(C2CC(C)=C(C)CC2)=O)COC(C)(C)CN1C(=O)C(=O)NCC(F)F 2622,C1(NC(C(C(COC)C)C)=O)CC2CCC1N(c1cc(C)nc(C3CC3)n1)C2 2623,c1(C(=O)NC2(C(N(CCC#C)CCOC)=O)CC2C)ncc(F)cc1F 2624,C1(OC(c2ccc(-n3cncn3)cc2Cl)=O)CCOC2(CCCC2)C1 2625,C12(NC(Cc3nc(C(C)(C)C)sc3)=O)CC1CN(C(C1CCC(C)(C)C1)=O)C2 2626,c1(C(N2CC(C(C(=O)NCc3c(CC)con3)OC)C2)=O)ncncc1C 2627,C(C)(CO)(C(=O)N1CC(CCNC(c2cnn(C)c2Cl)=O)(OC)C1)OC 2628,c1(C(=O)NCC(CC)NC(=O)C(C)C(C)CC)cc(C(=O)N(C)C)ccc1C 2629,c1(C(N(CC(CNC(CCOCCOCC)=O)C)CC)=O)cnn(CC(C)C)c1C 2630,c1(C(N(C(C)CNC(=O)C(F)OC(F)(F)F)C)=O)cccc2ccc(O)nc12 2631,C(=O)(CCN=c1[nH]c(=NC(C)c2ccc(Cl)cc2Cl)c2ccccc2[nH]1)NCC 2632,c1(OC)ccc2c(n1)NC(C(N1CCC(NC(C)=O)C(CO)CC1)=O)C2 2633,c1(C(N(CCNC(CCN(C(C)=O)C)=O)C2CC2)=O)ncc(F)c2ccccc12 2634,N1(C(C(C=CC)O)=O)CC(F)(F)CC1CNC(=O)Cn1cc(C)cn1 2635,Cc1cc(C)c(C(=O)NC2COCCC2NC(c2conc2C)=O)c(O)n1 2636,C(C(=O)NC1CCN(C(=O)C=Cc2ccc(C)o2)CC1C)(C(F)(F)F)OC(C)=O 2637,CC(O)CCCCCC(=O)NC1CCN(C(=O)CC2CCCCCC2)C1 2638,CC1(C)CCN(C(c2cnc(N)c(Cl)c2)=O)CC1NC(=O)Cc1n[nH]cc1Br 2639,C(=O)(C1CCCCc2ccccc21)NCCN(C(=O)C(C)C#N)CC 2640,C1(C(=O)NCCNC(C2C(CC(C)C)C2)=O)CN(CC(F)(F)F)CCO1 2641,c1(CCNC(C(=O)NC(C(F)(F)C(F)(F)F)SC2CC2)=O)cc2ccccc2[nH]1 2642,C(=O)(CC(C)C(=O)O)N(CCn1cc(-c2ccc(F)c(F)c2)nn1)CC 2643,C(=O)(CC1=CCCC1)NC1CC(C)(NC(C2(Cc3ccccc3)CCOC2)=O)C1 2644,c1(C(=O)Nc2scc(-c3c(CC)cc(F)cc3)n2)n[nH]c2c1CN(C)CC2 2645,C1(C(=O)NC2C(CNC(c3n(CC)ncc3Cl)=O)CC2)CC2(CCOCC2)C1 2646,N1(C(C2CCC(C)(C)OC2)=O)CC2CCCC2C1C(N1CC2CSCC(C2)C1)=O 2647,C1(CNC(CCNC(=O)OC(C)(C)C)=O)CCN(C(=O)Cc2ccoc2)C1 2648,C(CCC)(C(=O)NCCCN(C(C1CC1c1ccn(C)n1)=O)CC)=CCC 2649,C=C(C)C(C)(O)C(=O)N1CCCC(C)(NC(c2cccc(CC(F)(F)F)c2)=O)C1 2650,N1(C(C2(NC(C(CC(C)(C)C)OC)=O)CCSC2)=O)CCC2(COC(=O)N2)C1 2651,C(C(=O)NC1(CO)CC2(CCC2)C1)(C1=NOCC1)N(CCCN(C)C)CC 2652,C12(CNC(CSCC(C)C)=O)CCC(CC1NC(c1ccc(O)cc1F)=O)C2 2653,c1(C(=O)NCC2COCC2NC(C2CC2C2CCC2)=O)nccc2[nH]ccc12 2654,C12(COC)CC(C(=O)NCC(C3CCC3)NC(=O)CC3CCS(=O)(=O)C3)(CO1)C2 2655,C(=O)(C1CCCc2nncn21)NC1C(C=C)CN(C(C2(n3cnnn3)CC2)=O)C1 2656,C=C1CCC(C(=O)NC(Cc2ccoc2)C(=O)N2CC(C3CCCO3)C2)CC1 2657,Cc1cc(F)cc(C)c1C(N1CC2CCC1CN2CC1CCS(=O)(=O)CC1)=O 2658,c1(CC(N2C(CC)C(NC(=O)C(C)CSC)CC2)=O)ccc(C)cc1C 2659,N1(C(CNS(CC)(=O)=O)=O)CC(C)(NC(=O)CC(C2CCC2)C2CCC2)C1 2660,CC1=C(C(=O)NC2CC2NC(=O)CNC(=O)CC2CCCC2)CCS1(=O)=O 2661,CC1(NC(=O)CCCc2c(F)cccc2Cl)CCCN(C(=O)CNS(C)(=O)=O)C1 2662,C#CC1(O)CC(C(=O)NC(C)C=CC(=O)NCc2nncn2CC)C1 2663,C(=O)(C1=NNC(=O)C1)N1CCC(CNC(=O)C=Cc2ccccn2)(CO)C1 2664,c1(NC)cnc(C(N2CCC(C)(CNC(c3ncccc3C3CC3)=O)C2)=O)nc1 2665,C1(C(=O)NC(C(=O)NCc2n(C)cnn2)C2CC2)CC(=O)CCO1 2666,CC1(C)CCN(C(=O)CCC2CCOC2)C1C(N1CCOCC1C1CC1)=O 2667,C1(F)(C(=O)NCC2C=CC(NC(C3CCN(c4ncco4)C3)=O)C2)CCCCC1 2668,N1(C(c2cccc(C(=O)OC)n2)=O)CCC(NC(C2(CCO)CC2)=O)C(O)C1 2669,c1(C(=O)NC2CCCN(C(C=C(C)C(C)(C)C)=O)CC2)c[nH]c2c(F)cccc12 2670,C1(C(=O)NC2CC3CN(C(c4ccc(C#N)cn4)=O)CC32)CCCCC1C1CC1 2671,N1(c2cc(NCC3CSC3)nc(C)n2)CCC(C)C(C)(C)C1 2672,C1(N(C)C(=O)NCC2CCc3c[nH]nc3C2)CCc2cn(C)nc2C1 2673,c1(OCCNC(=O)NC2C(=C)COC2)ccccc1F 2674,c1(C(=O)NCC2(C)CCN(C(CC(=C)C)=O)C2)cc(OC)cc(Cl)c1F 2675,C1(C(N(c2cnn(C)c2)C)=O)CCCCCCN1C(c1cnn(C)c1Cl)=O 2676,c1(CNC(C2ON=C(CC)C2)=O)n[nH]c2c1CN(C(=O)C(C)(O)COC)CC2 2677,c12ccc(cc1)CC(=O)N2CCOC.C(C(=O)OC1CC1)OC 2678,C1(NC(c2n(C(C)C)ncc2)=O)CCCC(NC(=O)C(C)(C)c2cnc[nH]2)C1 2679,C(C)(CO)(C(F)F)NC(CN(CCC)C(c1nc(CC)oc1C)=O)=O 2680,C(=O)(CCC(=O)NC(c1ccccc1)CNC(=O)CSCC1CCCCO1)OC 2681,N1(C(CC(C)OC)=O)CCCC12CCN(C(=O)CC1(C)CCCCC1)C2 2682,C1(C(C)C)C(C(C)C)CN1C(=O)C(C1(O)CN(C(C2(F)CCC2)=O)C1)F 2683,c1(CC)ccsc1C(=O)NCC1(F)CC(NC(c2cc(C)cs2)=O)C1 2684,C1(NC(C2CCC(C)CN2C(c2c[nH]c(C(N)=O)c2)=O)=O)CCn2nnnc2C1 2685,CCCC(O)CC(=O)NCC1CC1CNC(=O)CN(CC(C)(C)C)C 2686,N1(C(C2(CNC(C(C)C3CCCC3)=O)CC23CCC3)=O)CCC2(CCCCC2)C1 2687,Cc1cc2[nH]c(C(=O)NCC3CC3NC(c3ccc(Br)c(N)n3)=O)cc2o1 2688,C1(NC(CCOCC#C)=O)CCCCC12CCCN(C(c1ccc(C)o1)=O)C2 2689,C(CC(C(C)(C)C)NC(c1c[nH]ccc1=O)=O)N(C(=O)CC1(C(F)(F)F)CC1)C 2690,C=C(C)CCC(C)OC(c1ccc(-c2ccncc2C)s1)=O 2691,c1(C(C)=O)ncc(C(N2CCC2CNC(=O)CC(C)c2ccco2)=O)s1 2692,C(CN=c1nc2ncn(C)c2c(NCCC(COC)OC)[nH]1)N(CC)CC 2693,C1(c2ccn(C)n2)CN(C(=O)CCCCN)C(C)(C)C1 2694,c1(C(=O)NCC2(NC(C(C=C=C)C)=O)CC(F)(F)C2)ccc2nonc2c1 2695,C1(CNC(=O)C=C2CCC2)CCCCC1NC(=O)C(=O)NC1CC1 2696,C12(C(=O)NCC3(CCNC(c4cnc(SC)[nH]4)=O)CC3)CCC(CC1O)C2 2697,C(C(O)C(=O)N1CC(O)CO1)NC(C1Cc2nccn2C1)=O 2698,Cc1cc(S(=O)(=O)NCC(=O)OC(c2ccccc2)c2ccco2)cc(C)c1Cl 2699,C1(N(C(COc2cn(C)nc2)=O)C(C)(C)C)CN(C(=O)Oc2ccncc2)C2CC12 2700,N1(C(C2C(=C)C2)=O)CCOCC(NC(c2cnc(C)c(CC(C)C)c2)=O)C1 2701,N1(C(C(C)CC2CCC2)=O)CCN(C(N2CCN(C(=O)C3=CCC3)CC2)=O)CC1 2702,C(C)(C(C(=O)N1CC(O)CC1CNC(=O)C(c1ccccc1)=O)N(C)C)OC 2703,C1(F)(CNC(c2ccc(CC)nc2)=O)CCC(CNC(=O)Cc2ccsn2)CC1 2704,C1(NCc2ccccc2C(N2C(C)C(C)(C)C2)=O)(CO)CC2CCCC12 2705,c1(C(=O)NC2CCC(NC(C(COC)OC)=O)C2)nn(C)cc1C 2706,C(C(C)(CC)C(=O)NCC1CC1C(C)C)NC(CC(=C=C)C)=O 2707,Nc1cc(Cl)c(Cl)cc1C(N1CC2C(CNC(c3ccnnc3)=O)C2C1)=O 2708,O=C(C1=CCCOCC1)NCC1CC2CCCC2N1C(c1cc(C2CC2)on1)=O 2709,C12(CNC(c3c(CC)nc[nH]3)=O)CCCC(CN1C(=O)C1=NOC(C)C1)C2 2710,C1(C(N(C2CCN(C(C3CS(=O)(=O)C3)=O)C2)CCCOSC)=O)CCN(S(C)(=O)=O)C1.S 2711,C1(OC)CN(C(=O)Cc2c[nH]nc2C)CC1NC(=O)CNC(c1cccnc1)=O 2712,Cc1cc(C(F)F)oc1C(=O)NCC1(CNC(C2CC3CCC2C3)=O)CC1(F)F 2713,c1(OCC)cccc(C(N2CC(O)(CNC(C3CCC3C(F)(F)F)=O)C2)=O)c1N 2714,C(CC)(C(=O)N(CCCNC(c1nsnc1O)=O)CC1CCCC1)=C(C)C 2715,C1(O)(CNC(c2nc(C)oc2)=O)CCCN(C(=O)CN2CCOCC2=O)C1 2716,C1(NC(c2c(CC)cccn2)=O)CN(C(=O)COc2ccsn2)CCC1CO 2717,c1(C(=O)NC(COC)CNC(c2coc(Cl)n2)=O)cc(O)cnc1Cl 2718,C1(NC(c2cnsc2)=O)CC2(NC(c3nc[nH]c3C(F)(F)F)=O)COC1C2 2719,N1(C(C2(N(C(C3CC(CC)OCC3)=O)C)CC2)=O)CCCC(C)(CO)C1 2720,CCCC(C)C(=O)NC1(COC)CN(C(=O)CC2(C#N)CC2)C1 2721,c1(C(N2CCC3(C(NC(C4C(=C)C4)=O)C3)CC2)=O)cc2cncn2c(O)n1 2722,N1(C(C(c2cccc(C)c2)C)=O)CC2CC(NC(c3c(C)n[nH]c3C)=O)C2C1 2723,C(=O)(CC(F)(F)C(F)(F)F)NCCC(C)NC(C1CC1(Cl)Cl)=O 2724,N1(C(C2C(c3cn(C)nc3)C2)=O)CCN(C(c2ccc(=N)[nH]c2Cl)=O)C(CF)C1 2725,c1(C(C)NC(C2CC3C=CC2C3)=O)cccc(NC(=O)CSc2nnc(S)s2)c1 2726,CCCC(C(O)C(=O)N(CCS(N)(=O)=O)C)NC(c1ncc(C)cc1F)=O 2727,C1(CNC(CCC=CC)=O)COCCN(C(c2cnn(C)c2C)=O)C1 2728,CC(C(=O)NCC1(C)CCCN1C(c1n[nH]cc1Br)=O)P(C)(C)=O 2729,C1(C)(CNC(=O)NCC2(NC)CCCC2)COCC(C)(C)O1 2730,C1(C(N2CCC(O)(CN(C(C3(CC)CC(C)(C)C3)=O)C)C2)=O)CC2C=CC1CC2 2731,C1(COC)CC(O)CN1C(=O)C(c1ccc(F)cc1)NC(=O)OC(C)(C)C 2732,CCCC(C)(O)C(=O)N1CCC(NC(c2cccc(CSC)c2)=O)C1 2733,C1(CNC(C=C(CC)CC)=O)CC2CCC1N2C(C12CCC(OC)(CC1)C2)=O 2734,Cc1nc(C)c(C(=O)NCC(O)CNC(=O)Cc2nccs2)o1 2735,N1(C(COCCC=C)=O)CCCC(C)(NC(=O)C(C)Oc2ccccc2C#N)C1 2736,C1(NC(CS(N)(=O)=O)=O)CC12CCN(C(=O)CC1(c3ccccc3)CCC1)CC2 2737,C1(CN(C(=O)Cc2cn(C3CC3)cn2)C)CCCN(C(c2cnc(Cl)n2C)=O)C1 2738,c1(C(=O)NCC(CNC(c2n(CC)ncc2)=O)O)cc(C(F)F)cc(C)c1 2739,Cc1c(C(=O)N(CCNC(C2CC23CCC3)=O)C2CC2)cncc1Br 2740,C(=O)(N1OC2C=CC1CC2)c1nc(CCNC(CCC2N(C)CCC2)=O)oc1 2741,Cc1ncnc(C)c1NC(C1CCOC1CNC(=O)CCc1cnn(C)c1)=O 2742,c1(C(N(C(c2cnc(CCOC)s2)C(=O)NC2CC2)C)C)ccc(C)cn1 2743,C1(C(=O)NCC(C)(C)CO)CCCCCN1C(=O)C(F)n1ccnc1 2744,C(N=c1ccc2c([nH]1)CCC2=O)C1C(C)CCCN1C(c1ccco1)=O 2745,N1(C(CC(C)(C)N(C)C)=O)CCC(C2CCCN(C(=O)Cc3c[nH]nc3O)C2)C1 2746,C1(NC(CSCC(C)C)=O)CN(C(C2(C#N)CCCC2)=O)CC(C)(C)C1 2747,S(=O)(=O)(c1ccc(F)cc1C)N(c1cc(SC)nc(C)n1)C1CCNCC1O 2748,C(=O)(N(OC)C1CCC1)C1N(C(c2ccc(CC)cc2)=O)C2C(C1)C2 2749,N1(C(C2CC(OC)C2)=O)CCCOC(C(C)C)C1.C(C)(C)(CN1CCCC1)NC=O 2750,N1(C(C(C)OCC#C)=O)CCCCC1CNC(=O)CC(O)C1CCCC1 2751,c1(COC)nc(C(=O)NC(C)(CNC(C2(CO)CC2(F)F)=O)CO)co1 2752,C(=O)(CC(O)C(Cl)(Cl)Cl)NC(CC)CNC(=O)C(CC1CC1)OC 2753,C1(OC)CC(C(=O)NCc2ncon2)N(C(c2ccc(Br)cn2)=O)C1 2754,N1(C(c2c(CC)cns2)=O)CCCCC1CN(C(=O)CN1CCC(C)C1)C 2755,c1(C(=O)NC2CC2CNC(C2(F)CCC2)=O)c(Br)ccc2ccccc12 2756,CC1CCc2sc(C(=O)NCCCNC(=O)C(c3ccc(F)cn3)(F)F)cc2C1 2757,C(=O)(C1=CCSC1)N(C1CCN(C(=O)C(O)C2CC2)C1)CCC 2758,S(=O)(=O)(c1cnc(-c2cccc(-c3c(C)ccc(Cl)c3)c2)s1)NC(=O)C(C)(C)Br 2759,C1(CC(N2C(CNC(=O)C(C)C3CCCO3)CC(OC)C2)=O)CC2(CCCC2)CO1 2760,c1(CNC(C2CSCCN2Cc2ncco2)=O)cc(Cl)ccc1O 2761,c1(C(N2CC(OCCNC(CN3CCC(C)CC3)=O)C2)=O)ccc(F)nc1F 2762,c1(OC)cc(-c2ncsc2C(=O)NC(c2cccnc2)C(C)C)c(F)cn1 2763,Cc1nc(C(=O)N(CCCN(C(=O)C(O)C2CC2)C)C)c(Br)s1 2764,C(=O)(C(C)C(C)NC(=O)CCn1cccn1)NC(c1nc(C)on1)(C)C 2765,C#CCCCCCCC(=O)N1CCC(C(C)C(N2CC=CC2CF)=O)CC1 2766,C1(N(C)C)(C=O)CCCC1.C(=O)(CCNC(c1ccsc1)=O)NC(CC)C1CC1 2767,c1(N2CC(O)(C(C)NC(CC(C(C)C)O)=O)C2)ccc(S(=O)(=O)N(C)C)cn1 2768,N1(C(c2c(C)cc(CO)o2)=O)CCN(C(=O)C=Cc2cc[nH]c2)C2CCCCC12 2769,Cc1cc(Cl)ccc1OCC(=O)NCCC(C)N(C)C(C1COC(=O)N1C)=O 2770,Cc1c[nH]c(C(=O)NC2CCC(CNC(=O)Cc3cc(Br)cs3)CC2)c1C 2771,Cc1c(C(=O)NC(C)(C)CNC(=O)C(F)CC2CCCC2)cccc1N 2772,c1(OC)ccc(S(=O)(=O)N2CCC3CN(Cc4cccc(Cl)c4Br)CC23)cc1 2773,C#CCC(C)C(=O)N1CCCC1C(C)(C)NC(=O)Cn1ncccc1=O 2774,Cc1coc(C)c1C(=O)Nc1ccccc1.N12CC3C(C3C1)c1cn(nn1)CC2 2775,N#Cc1ncc(CN2CCC(Cn3cc(-c4sccc4Br)nn3)C2)s1 2776,Cc1nn(C(C)(C)C)cc1C(=O)NC1CCN(c2cccnc2)C1 2777,CCC(CC)C(=O)N1CCC1C(=O)Nc1cnn(CCO)c1 2778,Cc1c(O)ccc(C(N2CCC(NC(C3COCCN3C)=O)C23CC3)=O)c1C 2779,C(=O)(C(F)C1CC(N(C(=O)CON2CCCC2)C)C1)N(CC(=O)OC(C)(C)C)C 2780,CC1CN(C(c2cnc[nH]2)=O)CC(C)C1NC(c1scnc1Cl)=O 2781,Cc1ccc(C=CCC(N2CCC(CNC(=O)CC(C)O)C2(C)C)=O)cc1 2782,C(CC)(CCCC(=O)N1CCCC(C#N)C1)NC(CCCCCC)=O 2783,C12(C(=O)OC)CC(C(=O)N(CCCN(C(=O)CSc3n[nH]c(O)n3)C)C)(C1)C2 2784,N1(C(COCC)=O)C(CNC(c2nocc2C(C)(C)C)=O)CC2CCCCC12 2785,c1(OCC)sccc1C(=O)NCC(C)CNC(=O)C(C1CCOCC1)=O 2786,c1(C(N2CC3(CCN(C(C=CCCC)=O)C3)C2)=O)ccc(Br)c2cn[nH]c12 2787,C(=O)(C1=CN=C2N=CNN2C1)NC1(C)CCCN(C(C2(F)CC3(CCC3)C2)=O)C1 2788,c1(C(=O)NC2CC(n3cc(CCC4CCCO4)nn3)C2)ccc(Br)cc1 2789,C1(NC(c2cc(CC)no2)=O)C2CCC(C2)C1C(=O)Nc1cc(CO)cc(Cl)c1 2790,c1(C(C(=O)NCCN(C(=O)C=CC2CCCN2C)C)F)ccc(C(F)(F)F)cc1 2791,c1(C(=O)NCCC(C)N(C(C=CCCC=C(C)C)=O)C)c(C)ncnc1O 2792,C1(CC(=O)NC(=O)CN2CCCC2C(C2CC2)CC2CC2)CCCC12CC2 2793,N1(CC(N2CCC(C(C)(C)NC(C(CC=CC)C)=O)C2)=O)OC(C)(C)CC1=O 2794,C1(CCCNC(CCCC)=O)CCN(C(=O)C(C)(C)Oc2ccc(Cl)cc2)CC1 2795,c1(C(=O)OC)cc(NC(=O)C(C)n2ccnc2)cc(Cl)c1 2796,c1(COC)nc(NC2CC(C)SC(C)C2)cc(N2CCN(c3ncc[nH]3)CC2)n1 2797,c1(C(N(CC(C)NC(=O)CN2CC=CC2)C)=O)cn2c(n1)CCC2 2798,c1(C(N(C)CCNC(c2cccn2C)=O)=O)cc(F)cc(F)c1 2799,C1(C(=O)NCCc2c(CNC(C3(CC)CCOC3)=O)nco2)CN=C2N=CNN2C1 2800,C1(NC(C(CC)OC)=O)CCN(CCC2CCOCC2)CC1O 2801,C#CC1(C(=O)NCCC2CC(C)(C)C2)CCN(C(=O)CCC2CCCO2)CC1 2802,C12(NC(C3N(CC)CCOC3)=O)CCOC(CNC(=O)C(C3CC3)SC)(C1)C2 2803,CC(CNC(C1(CF)CC1)=O)(CO)NC(=O)C=CC(=O)OC(C)(C)C 2804,C1(NC(CNC(CC)=O)=O)CCC2(CC1)CN(C(=O)C=CCn1cncn1)CCO2 2805,N1(C(=O)CSc2nnc(S)s2)CC(C2CN(C(c3ncc(Cl)cc3F)=O)C2)C1 2806,Cn1cnc(C(C(=O)NCC2CCOC2)N(CCCCO)C)n1 2807,C(C)(C(CC(=O)NC(C)CCc1cn[nH]c1)NC(=O)CC1CCC=CCC1)OC 2808,C1(CC(N2CC(NC(C(C)(C)OC)=O)CC2(C)C)=O)CCc2ccccc2C1=O 2809,c1(OCC(=O)NCC2(F)CCC(NC(c3ccc(CO)o3)=O)C2)cccc(F)c1 2810,N1(C(c2nc(CCCC)sc2)=O)CCC2CN(C(c3cnc(C)cc3Cl)=O)CC12 2811,c1(NCCCc2n(CCC)ccc2)cnccc1C(=O)OC 2812,N1(C(c2cc(OC)n(C)n2)=O)CCC(C(N2CC(O)(CO)C2)=O)C12CC2 2813,c1(OC(CC)C)ccc(C(N2CCCC(CCNC(=O)CC(F)(F)F)C2)=O)cc1 2814,N1(C(C(N2CCOC2=O)C)=O)CCOC2CN(C(c3ncc(Cl)cn3)=O)CC12 2815,CCCCC(C)C(=O)NC1CC(CNC(C2(C(F)(F)F)CC=CC2)=O)C1 2816,C12(CNC(c3c(C)nn(C)c3)=O)CC(CCO1)N(C(=O)COC(C)(C)C)C2 2817,C1(F)(C(=O)NCC2N(C(CC(=O)NC)=O)CCC2C)C(C)(C)C1(C)C 2818,C(CCC(C)(C)NC(C1CCCN1S(C)(=O)=O)=O)NC(CN(CC(C)(C)C)C)=O 2819,CC1(NC(C23CC(CN2C(C2CN4CCC2C4)=O)C3)=O)CC2CCC1C2 2820,c1(C(N2CC3CCN(C(CCNC(C)=O)=O)CC32)=O)ccc2c(c1)COCCN2 2821,C(=O)(C(F)CC(C)(C)NC(=O)C1=NOC(C)C1C)N1CCC(COCC)C1 2822,CC(C)(CNC(c1cncs1)=O)CC(=O)NC1(CO)CC(F)C1 2823,CCC(C(=O)NC)NC(C1CC(O)(CNC(C2(C(=O)OC)CC2)=O)C1)=O 2824,N1(CCC)C(=S)NC(c2cc(C(F)F)no2)C=C1CCC(C)(C)C 2825,C(=O)(C(C)(C)CS(N)(=O)=O)NC1CCN(C(C2(Oc3cn(C)nc3)CC2)=O)C1 2826,CC1NC(=O)CCC1CNC(C1CC(NC(c2cn(C)c(=O)cn2)=O)C1(C)C)=O 2827,N1(C(c2c(OC)cc(Cl)cc2)=O)CCn2nnc(C(=O)NC3CCOC3)c2C1 2828,CC#CCCCC(=O)N1CCC(O)C(NC(C2CCCC(C)(C)C2)=O)C1 2829,CC(C)C(CO)C(=O)N(C(CNC(c1cnn(C2CC2)c1)=O)C1CC1)C 2830,C1(C(=O)NCC2(SC)CCC2)CN(C(=O)CCc2ccoc2)CCO1 2831,c1(CN2CC(CC(=O)NCc3nc(C)[nH]n3)OCC2)cccc([N+](=O)[O-])c1 2832,C1(O)(CNC(=O)Cn2cnnn2)CCCN(C(c2ccccc2SCCO)=O)C1 2833,c1(C(=O)NC2CCC(NC(c3c(Cl)ncc(C)c3)=O)C2)ccc2nc(O)[nH]c2c1 2834,C1(CN(C)C(C2CC3(CC3)C2)=O)CCCN(C(c2snnc2C2CCC2)=O)C1 2835,N1(C(C2C(=C)CC2)=O)C2CCCC1CC(CNC(c1c(Cl)ccc(F)c1N)=O)C2 2836,Cc1cccc(CC(c2ncc[nH]2)NC(=O)NCCc2ccccc2C)c1 2837,C1(CC(=O)NC(COC(C)=O)CO)CN(C(C2CC(OC)C2)=O)CC12CC2 2838,Cc1nn(CCO)c(C)c1C(=O)NCC1CC(CNC(=O)CN(C)C(N)=O)C1 2839,c1(NC(CN(C(CC2ON=C(C)C2)=O)CC2CC2)=O)ccc(C)nc1O 2840,CC(C(=O)N1OC2CCC1C2)C1CCN(C(C2(C#N)CC(F)(F)C2)=O)C1 2841,c1(-c2cnc(C)o2)nc(C(C)C)nn1CC(C)(C)O 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2878,C1(C#N)(C(N(CCCNC(=O)CCCN2CCCC2)C)=O)CCS(=O)(=O)CC1 2879,C(C(CNC(c1cnn(-c2ccc(Cl)cc2)n1)=O)C(F)(F)F)NC(C1C(C)C1)=O 2880,C12(C(=O)NC3C(CNC(=O)COc4ccc(Br)cc4)C3)CC1CCC2(F)F 2881,C1(C(=O)NC2CCCC(F)(F)C2)Cc2cc(O)ccc2CN1S(=O)(=O)CCCl 2882,c1(CNC(=O)Nc2ccc(-c3cnn(C4COC4)c3)nn2)ccc2c(c1)CCC2 2883,Cc1cc(=NCCc2c[nH]nc2O)[nH]c(=NCC2CCN2C(=O)OC(C)(C)C)[nH]1 2884,C(N=c1cc(C(C)=O)c([N+](=O)[O-])c[nH]1)C1C(C)CCN(C(C(CC)(F)F)=O)C1 2885,C1(C)(C(N(C)CC2CCN(C(CCC(=C)Br)=O)CC2)=O)CC(OC)CN1C 2886,C(=O)(C1c2c[nH]nc2CN1C(c1cc2ccccn2c1)=O)NCCOCCC#C 2887,CCCCC(CC)C(=O)NCCCN(C)C(C1CC1C(C)(C)O)=O 2888,C1(O)(C(N2CC(NC(c3nc(Cl)cs3)=O)CC(C)C2)=O)CN2CCC1CC2 2889,C1(C#N)(C(N2CC(COC)(CNC(=O)CCCc3ccsc3)C2)=O)CC1(C)C 2890,C#CC1CN(C(=O)CCCN(C)C)CC1OCC 2891,c1(C(=O)NC2C3CN(C(C=C(C)C(F)F)=O)C2C3)ccc(F)cc1C(F)(F)F 2892,c1(C(=O)NC2(COC)CN(C(C3CC(O)C3)=O)C2)cc(C2CC2)nc(O)c1 2893,C(=O)(CC1=NNC(=O)C1)NCC1(O)CCN(C(CCc2cc(C)on2)=O)C1 2894,C1(C)(C(N(CCN(C(C)C)C(C2CCC(F)(F)C2)=O)C)=O)CCCN1C 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2985,c1(OC)nc(C)cc(=NC2CC23CC(NC(=O)C(C)CC(N)=O)C3)[nH]1 2986,C1(C(=O)OCCCC2CCCC2)CC2(CCCC2)CO1 2987,c1(OC)cc(C(N2CCCC(NC(=O)CC3SC(=N)NC3=O)CC2)=O)cc(C)n1 2988,C#Cc1cncc(NC(=O)CC23CCC2CN(C(=O)C(C(C)C)NC(C)=O)C3)c1 2989,CN1CC(C)(C(N2CC3(CCN3C(C3CSC3)=O)C2)=O)CCC1=O 2990,N1(C(c2ccc(C)nn2)=O)CCN(C(=O)CCC2(C)CC2)C(C(F)F)C1 2991,N1(C(CP(C)(C)=O)=O)CC2C3CCC(C2C1)N(C(=O)C=C1CN2CCC1CC2)C3 2992,C(=O)(C1CCCc2nn[nH]c21)NCC1(NC(c2ccc(Cl)c(O)c2)=O)CCOC1 2993,Cc1ccc(C(N2CCCC(C3(NC(c4cncs4)=O)CC3)C2)=O)c2c1CCC2 2994,N1(C(CCCC#CC)=O)CCC2(CCC2NC(=O)CC2OCCC2(C)C)CC1 2995,c1(C(=O)OC)cc2oc(C(N3CCC(O)(CSC)C3)=O)cc2[nH]1 2996,N1(C(C2C(C)(C)COC2)=O)CCN(C(=O)Cc2cnsc2)CC(O)C1 2997,CC1CCCC(C(=O)N(CC(=O)N(C2CCOC2)C2CC2)CC2CC2)CC1 2998,N1(C(C(CC=C)C(C)C)=O)CCC(C2CN(C(c3ccc(O)nn3)=O)C2)C1 2999,C1(C(=O)NC2(C(=O)NCC)CC2)C2CC3C(C2NC(=O)C(C)COC)C13 3000,Fc1ccc(C(c2nnnn2CC2CC2)NCc2nncn2C2CC2)c(F)c1Br 3001,Cc1nc(CSCCC(=O)NC2CCCC2NC(c2cnc(C)s2)=O)cs1 3002,CC1CCC(C)C1NC(c1c(CNC(=O)CN=[N+]=[N-])nnn1C)=O 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3021,c1(C(N(C2(C(=O)NC(C3CCCC3)C#C)CC2)C)=O)ccc(N)cc1C 3022,n1(CC#C)cc(CNC(=O)C(C)N(C(=O)C=CCN2CCC2)CC)cn1 3023,C(=O)(C(F)(F)C(O)C1CC1)NC1CC2C(NC(C3(C(N(C)C)=O)CC3)=O)C2C1 3024,N1(C(C(=O)NCCNC(C)=O)=O)CC=C(c2cccc(Cl)c2C)CC1 3025,C(=O)(CCCC(=O)N1CC2CC2(NC(C2CCC3CCC2O3)=O)C1)NC(C)C 3026,CN=c1ncc(-c2ccc(F)c(CN3CCC(N(C)CC4CC4)CC3)c2)c[nH]1 3027,C1(C(C)NC(C2(C(=O)NC)CCC2)=O)CCCN(C(c2sc(C)cc2Cl)=O)C1 3028,Cc1c[nH]cc1C(=O)NC(C1CC1C(=O)NCCC(C)(C)C1CC1)C 3029,c1(CC)[nH]nc(C(N2CC(NC(C3CCCN3C(=O)NC)=O)C(SC)C2)=O)c1Cl 3030,Cc1nc2c(cc1C(=O)NCCC1COCCN1C(=O)C=C1CC1)c(C)nn2C 3031,C1(C(N(CCN(C(Cc2cc(CC)no2)=O)C)C)=O)CC12CCC(=O)CC2 3032,Cc1ccc(NC(C2C(NC(=O)CCN=[N+]=[N-])C2(C)C)=O)c(C)n1 3033,C(C(=O)NC1(C2CCCN2C(c2nccnc2N)=O)CC1)(C(C)C)SCC 3034,C(=O)(C(O)CC(C)(C)C)NCC(CNC(CC(C)(C)OC)=O)C 3035,CCCCC(O)C(C)C(=O)NC(C)C=CC(=O)NCCC(C)C(F)F 3036,c1(OC)c(F)cc(C(=O)NC(C2CCCC2)CNC(=O)C(F)OC)cc1Cl 3037,N1(CC=O)CC(C)(C)C12CCOCC2.c12cc(cc(C)c1)N(C)CCC2.CS 3038,C#CCCC(O)C(=O)NC(C)CCNC(c1snnc1CC)=O 3039,C1(C(N2CCCC(NC(CCc3ncc(C)[nH]3)=O)C2C)=O)CS(=O)(=O)CC(=O)N1 3040,C(=O)(CCCCC#N)NCC1N(C(COCC(=C)C)=O)CC(O)C1 3041,N1(C(CC)C(C)C)CC2COCC2(C(=O)NC2CCN(C3CCCCC3)C2)C1 3042,CCC(C)C(=O)C(=O)NOCC(=O)NC1CC(O)C(O)C1 3043,N1(C(C(C(CC)C)N(C(=O)CN2CCCCC2)C)=O)CCN2CC(O)CC2C1 3044,N1(C(c2c(N(C(C)C)C)cccc2)=O)CC2CN(C(=O)C(C)(C)F)CC2(C)C1 3045,C1(C(=O)NC(c2ccn(C)n2)C(N2CC(SC)C2)=O)OC2CCC1C2 3046,CC1C(C)C(C)CN1C(=O)C(=O)Nc1ccc(OCC(=O)N(C)C)cc1 3047,CCC(CCC(=O)NCc1ccon1)NC(=O)Cc1cn(C)nc1C 3048,Cc1cc(=NC(=O)C(=O)Nc2ccc(C3OCCO3)cc2)[nH]n1C(C)(C)C 3049,c1(C(N(CCNC(C2CCCC2n2cccc2)=O)CC)=O)ncc(C)cn1 3050,CC(C)CC(F)C(=O)NC1CCCN(C(=O)CCN(C)C(=O)OC(C)(C)C)C1 3051,C(CC(C)C)(C(=O)NCC1(N(C)C)CCC1)ONC(COC(CC)CC)=O 3052,c1(CCNC(C)=O)ccc(C(=O)NCC2C(NC(=O)CCCF)C2(C)C)cc1 3053,c1(C(N(CCNC(C(n2c(C)ncc2)C)=O)C2CC2)=O)c[nH]c(=S)cn1 3054,CCCC(C)CC(=O)N(CCCC(=O)NCCOC1CCOC1)C 3055,c1(C(=O)OCCC2CCC(C)C2)ccc(SC(F)F)cc1 3056,C(=O)(CC1OCc2ccccc21)N(CCNC(C(=O)NCC)=O)C(C)C 3057,Cc1nnc2n1CCN(C(C1CCCN(CCS(C)(=O)=O)C1)=O)C2 3058,c1(C(N2C3CCC(CNC(C4C(=C)CC4)=O)(C3)C2)=O)cccc2ccn(C)c12 3059,CC1CN(C(=O)Cc2cc(Cl)ccc2O)CCC1N(C(=O)Cn1ccnn1)C 3060,N1(C(c2cnn(C)c2C)C(=O)NCCCSCC)CC(C)CCCC1C 3061,C1(C(=O)NCC(CC)N(C)C)(CNC(c2cc(Cl)c[nH]2)=O)CCCC1 3062,C(C(CC(C)C)C(=O)NC(C)Cc1nc[nH]n1)NC(c1c(C)noc1)=O 3063,c1(C(N2CC(CC=C)(NC(C3CC3CF)=O)C2)=O)cn2cccc(C)c2n1 3064,C12(NC(c3cncc(-n4ccnn4)c3)=O)CC1CN(C(C1CCC13CCC3)=O)C2 3065,N12CC3(CC(F)(C1)C3)CC2=O.C1(NS(C)(=O)=O)CC(NC(=O)Cc2ccon2)C1 3066,CN1C(=O)CC(C(N2CC(C(N)=O)(CNC(=O)CNC=O)C2)=O)C1c1ccnn1C 3067,S(=O)(=O)(c1ccc(F)cc1)N(CC(=O)N(CCNC(C(C)O)=O)C(C)C)C 3068,C(=O)(CC(C(F)(F)F)c1ccon1)N1CC(O)(CNC(C(C)(C2CC2)OC)=O)C1 3069,N1(C(C=C(COC)C)=O)CCC(N(C(=O)COC2CC2(F)F)CCO)C1 3070,c1(OC)ccccc1C=CC(=O)N(C)CCNC(=O)CC(c1c(C)noc1C)C 3071,C1(NC(C=CCC(C)(C)NC(=O)CC2(O)CCOCC2)=O)CC2(CNC(=O)O2)C1 3072,CC1CCN(C(c2cc(Cl)c[nH]2)=O)C(C(=O)NCc2nccn2C)C1 3073,Cc1cc(CNC(C2(O)CCN(C(C3CCCN(C)C3)=O)C2)=O)cc(O)n1 3074,C1(CNC(C(C=CCCC)O)=O)CN(C(=O)C(C)(C)CF)CCO1 3075,C(C(O)CN=c1[nH]c(C2CCCC2)nc(=N)[nH]1)NC(c1c(S(C)=O)cccc1)=O 3076,C(N=c1[nH]nc(-c2cccnc2)s1)C1CCC(NC(c2cc(C)ncc2)=O)C1 3077,c1(N2CC(CNC(Cc3cccc(C)c3C)=O)OCCC2)nc2cccc(C)c2o1 3078,Cc1nn(CC(=O)NCC2CCC2NC(=O)CC=CC(C)(C)C)c(C)c1C=NO 3079,N1(C(Cn2c(C(=O)OC)cc(C)n2)=O)CCC(F)C(NC(c2sccc2Cl)=O)C1 3080,CC1CCN(C(c2cncnc2)=O)CC1N(C)C(C1CCCCCC1)=O 3081,N1(C(CCCCCOCC)=O)CCC2CCN(C(=O)C(C(C)C)C(C)C)CC12 3082,C(=O)(C(C)(C)CN(C)C(C1COCC(C)O1)=O)N(CC(CC)OC)C 3083,c1(NC2C(NC(C=CSC)=O)CCCC2)ncnc2scc(Br)c12 3084,c1(OC)cc(Cl)c(Cl)cc1C(=O)NC12CCN(C(=O)OC(C)(C)C)CCC1C2 3085,Cc1cccc(OCC(N2CCC(NC(=O)CCCF)C2C)=O)c1C 3086,c1(NC(C2C(NC(c3cccc(C)c3)=O)C2)=O)ncnc2[nH]c(C)cc12 3087,C1(CNC(c2cnc(O)s2)=O)CN(C(C2C(F)(F)C23CC3)=O)CCCO1 3088,c1(C(=O)NC(CNC(CCCCC)=O)CC(C)C)cc(C2CC2)ccc1F 3089,C(C(CC(C)C)C(=O)NCC1(C)CNC(=O)O1)NC(C1(CC=C)CC1)=O 3090,C1(CC(C)NC(=O)CSC(F)F)CCN(C(=O)COc2ccc(CO)cc2)CC1 3091,c1(C(=O)NC2CC(N(C(C=CSC)=O)C)C2)ccc(NC(=O)N(C)C)cc1 3092,N1(C(C2C(CC(C)C)C2)=O)CCCC1CN(C)C(C1(CCCO)CCCC1)=O 3093,C1(C(N2CC(O)(CNC(c3ccc(CO)o3)=O)C2)=O)CCCC12CCC2 3094,N1(CC(=O)NC(CNC(C2C(C)OC(=O)N2)=O)C(C)(C)C)CCC(=O)NC1=O 3095,C1(CC(=O)OCC)CCCC2CN(C(=O)C(N)CN3CCCC3=O)CC12 3096,CC1CC(C)(C(N2CCCC(C)(CNC(=O)CC3CCNC3=O)C2)=O)CC(C)O1 3097,c1(C(CCC(=O)NC2(C(c3ccc(OC)cc3)O)CC2)C)c(C)cc(C)cc1C 3098,c1(C(N(C2CCN(C(C3CCCC4CC34)=O)C2)CC)=O)ccc(Cl)c(Cl)c1 3099,c1(OC)nc(C)cnc1C(=O)NCc1cccnc1CNC(=O)CC(C)F 3100,c1(C(=O)NCc2c(CN(C(=O)C(C)(C)F)C)cccc2)cc(N)c(F)cn1 3101,C(=O)(CCCNC(=O)C1CC1)NC(CN(C(=O)CC1CC1(C)C)C)(C)C 3102,c12cccnc1C(=O)N2.C1(NC(N)=O)CCOC1C(N1CC(O)C1)=O 3103,N1(c2ncc(CC)cn2)CCOCC(NC(=O)Cc2noc(C)n2)C1 3104,c1(C(=O)NCC2CN(C(c3c(C)n[nH]c3)=O)C2)ccnc2c1ccn2C 3105,C(=O)(C(C(C)CC)N(C)C)NCCC(=C)CNC(c1cnccc1N(C)C)=O 3106,c1(C(C)C)cnc(C(N2CCC(c3n[nH]c(N(C)CCN(C)C)n3)CC2)=O)nc1 3107,Cc1ccnc(O)c1C(=O)NCC(C)NC(c1cn(C)c(-c2ccccn2)n1)=O 3108,c1(C(N2CCC(NC(C3CC(C)(O)C3)=O)C2C)=O)ccc(COC(C)C)cc1 3109,C1(CC(N2C(CC(=O)N(C)Cc3ncn(C)n3)CC2)=O)CCCC2CC12 3110,N1(C(c2ccc(CC)s2)=O)CCC2CC2(NC(=O)CCS(N)(=O)=O)CC1 3111,C1(NC(C(C2CCCC2)OC)=O)CCNC1(C)C 3112,c1(N2C(CNC(C3N(C(C)C)CCC3)=O)C(C)CC2)nc(Cl)ncc1C(F)(F)F 3113,N1(C(C(C)(O)C2CCC2)=O)CC2CC(C1)C2NC(c1sc(Cl)cc1Cl)=O 3114,C1(CNC(CCCC)=O)C(C)CCCN1C(c1ccc(CC(C)C)nc1)=O 3115,c1(C(=O)NC2CCCC(CN(C)C(c3cnsc3)=O)C2)ccc2c(c1)CCCS2 3116,N1(C(C)=O)CCCC2C1CCCN2C(c1ccccc1NC(c1ccco1)=O)=O 3117,C1(C(N2CC(c3cn(-c4c(OC)cccc4)nn3)C2)=O)CCC(C)(C)OC1 3118,c1(C(N2C(CC)C(NC(c3ccccc3Cl)=O)CC2)=O)ccc2c(c1)N(C)CC2 3119,n1(C(CCCC)C)c(-c2ccc(Br)c(Cl)c2)csc1=Nc1cccc(Cl)c1OC 3120,C1(NC(CC2(C=C)CCC2)=O)CCN(C(=O)CC2CC(=O)C2)C(C)C1 3121,N#Cc1cc(C(N2CC(NC(C3CCSC3)=O)C(C=C)C2)=O)cc(F)c1F 3122,C12(CNC(c3c(Cl)ccc(N)c3)=O)CCCCC1CN(C(=O)Cc1ccoc1)C2 3123,CN1CC(NC(C2CN(C(=O)CN3CCNC3=O)CC23CC3)=O)CCC1=O 3124,C1(NC(C(c2ccc(Cl)cc2)C)=O)CN(C(=O)C(c2cccnc2)=O)CC12CC2 3125,CCC(C)(C)C(C)CC(=O)NCC1CC(NC(c2ncc3[nH]ncc3n2)=O)C1 3126,CCCC(C)C(=O)N1CCCC1Cn1cc(CNC(=O)CSC(F)(F)F)nn1 3127,c1(OCC)cc(Cn2cc(-c3ccccc3C#N)nn2)ccc1Cl 3128,C1(C(N2CCCCC(CNC(C3(CC)CC3)=O)C2)=O)CC2CCC(C1)C2O 3129,c1(C(=O)NC(CC(C)NC(c2cc[nH]c2)=O)C)ccc(-c2cnc[nH]2)cc1 3130,N12CC3COCC3(C1)C2.N1(C(C(CC)Sc2cccs2)=O)CCC(=CCO)CC1 3131,C1(NC(C(C)C2(O)CCC2)=O)COCCC1NC(=O)C(C1CCOCC1)F 3132,C1(C(N(CC(CCC)O)C)=O)CC(OC)CN1C(=O)CC1CC2(CCC2)C1 3133,C1(N(C(C2CC(=C)C2)=O)C)CCCN(C(=O)C(C)(C)C(F)F)CC1 3134,C1(C(=O)NC2(CCCC)CC2)CCN(C(c2csc(O)n2)=O)C(C)(C)C1 3135,C(=O)(C(=O)CC(C)C)NCCCC(N1CCCC(CC=CC)C1)=O 3136,C(=O)(C(C)CC(C)CC(C)C)NCC1CC(NC(c2nnn(CC)c2C)=O)C1 3137,c1(CCC(=O)NCCN(C(c2cncnc2)=O)CC)ccc2c(c1)NC(=O)CO2 3138,C1(C(C)C)CN2CC1NC2=O.c1(COC(C)C(c2ccccc2)C)ccccc1 3139,C1(C(N2CC(C)C2C(=O)NCCc2cn(C)nn2)=O)CC12CCCCC2 3140,N1(CC(=O)NC2CC2)CCC(N(C(C2CC23CCOC3)=O)Cc2nncs2)CC1 3141,Cc1ncc(NC(=O)C(C)NC(=O)C(C)C2(O)CCC2)c(C)c1C 3142,C1(OC)CC2C1CCN2C(C12CCC(CC1NC(=O)CCC1CC1(F)F)C2)=O 3143,c1(CC)cc(C(=O)NC(C)C(C)NC(=O)C(F)C2CCCC2)ccc1O 3144,C(=O)(C(F)C(C)CNC(C1CCS(=O)CC1)=O)NCc1c(OC)nn(C)c1 3145,C12(NC(CCc3cnc(C)o3)=O)CC1CN(C(=O)C(C)OCC(C)C)C2 3146,N1(C(C=Cc2ccc(=N)[nH]c2)=O)CCC2CC(NC(=O)C(N)=O)CCC2C1 3147,c1(C(=O)OC)cn(C)nc1C(=O)NC(C)CNC(=O)Cc1cnns1 3148,Cc1nc2cc(NC(C3C(O)CCN3C(=O)CC3CCCCO3)=O)cnc2[nH]1 3149,c1cnc2c(c1)cc(NCC1CCN1C1CC1)c1cccnc21 3150,C1(CSC)CCN(C(=S)Nc2ccc(Cl)c(OC)c2)C1 3151,N1(C(=O)OC(C)(C)C)CCc2ccccc2C1CC(=O)OCC(F)F 3152,C1(C(=O)NC(C(N2CC(C)=C(C)C2)=O)CCN(C)C)CC2(CC(=O)C2)C1 3153,C1(CNC(Cc2scc(C)c2)=O)CCCN(C(c2cccc(OC(F)F)c2)=O)C1 3154,C1(NC(c2nc(OC)c(C#N)cc2)=O)CCn2c(C)cnc2C1 3155,C(=O)(CCCCCc1cn(C(C)CN2CCCC2)nn1)Nc1cc(C)nn1C 3156,Cc1ccc(C(=O)NC(C)Cn2cc(-c3cncs3)nn2)cc1[N+](=O)[O-] 3157,N1(C(CN(C2CCC2)C)=O)CC(NC(C2C=CC=CC=C2)=O)C(c2nccn2C)C1 3158,C1(C#N)(NC(CC(C)O)=O)CCN(C(=O)CN2C(=O)CSC2=S)C1 3159,CCCC(C(=O)NC1(C)CCN(C(c2nccn3ccnc23)=O)C1)C(C)C 3160,CC1(NC(c2cnc(Br)s2)=O)CCN(C(C2(O)CCC2)=O)C1 3161,CC(C)(C#N)CCCC(=O)NC1C2CN(C(c3n[nH]cc3C(F)(F)F)=O)CC12 3162,c1(CCNC(c2n(CC)ccn2)=O)cc(C(=O)OC)sc1Cl 3163,c1(OC)ccc(Br)cc1C(c1nnnn1Cc1ccco1)NCCc1ccns1 3164,c1(SCC(=O)NC(C)CC(C)O)ccccc1C(=O)O 3165,C1(CC(=O)NCC2CCN2C(=O)C=C2CCCCC2)CC2(CCC2)C1 3166,c1(OC)cc(NC(=O)C(CN=[N+]=[N-])NC(C2CCC(OC)CC2)=O)cc(O)c1 3167,c1(C(N2CCCCC2c2nc[nH]n2)C(=O)NCC(C)C)nc(Br)nn1C 3168,C1(CCC)CN(C(=O)Cn2nc(C)nc2C)CCN1C(=O)C1=C(Cl)CCC1 3169,N1(CC2N(C(C3CC3c3ccc(Br)cc3)=O)CCC2)CCN2CC(O)CC2C1 3170,C1(N(N2CCCC2)C(=O)OC(C)(C)C)CCC(NC(=O)CCc2ncc[nH]2)CC1 3171,C(=O)(C(C)(C)C(C)C)N1CC(CC(C)NC(C2C(C)=CCS2)=O)C1 3172,C1(NC(CC(C)N(C)C)=O)CC(C(=O)NCC2=CCCC2)C1(C)C 3173,C1(C(=O)NCCC(=O)NC(C)C)C(C)OCCN1C(c1cc(O)n(C)n1)=O 3174,C(=O)(C1=NN(C)C(=O)CC1)Nc1scc(-c2c(F)ccc(-c3ccc(OC)s3)c2)c1 3175,C(=O)(CCCCCF)NCCN(CCOC)C(C1CC1C1CCCC1)=O 3176,CCCC(C)(O)CC(=O)NC1(C)CCCCC1C(=O)NC(CO)CCF 3177,CC(CNC(c1csc(O)n1)=O)C(F)C(=O)NCCF 3178,N1(C(c2cnc(OC)s2)=O)CC2(CCC2NC(=O)C(O)Cc2cn(C)cn2)C1 3179,CCC(CC)(CCNC(=O)CC1CC1(Cl)Cl)NC(=O)C(O)C1CC1 3180,c1(OC)cccc(C(N2CC(NC(=O)CC(=O)Nc3nccs3)CC(C)C2)=O)c1Cl 3181,C1(CCNC(c2ccsc2)=O)CCCN1C(C1CCCN1C(=O)C(F)(F)F)=O 3182,N1(C(C(C)OC)=O)CCN(C(=O)C(C)CSC)C(C2CC2)C1 3183,N1(C(COCCCCC)=O)CC(CNC(=O)CC2CCCOC2)C(F)(F)C1 3184,N1(C(C(F)=C(C)C)=O)CCC2(CCCC2NC(c2cc(C)sc2C)=O)C1 3185,C1(C(C)NC(c2c(C(C)C)c[nH]n2)=O)CN(C(=O)CCCC2CC2)CCO1 3186,C1(C(=O)NC2C(CNC(c3c(C)[nH]cc3)=O)COC2)CCn2cncc2C1 3187,N1(C(C2CCCN(CC(C)C)C2)=O)CCCN(C(c2ncccn2)=O)C(CO)C1 3188,CC(C)C(O)C(F)(F)C(=O)NCCc1ocnc1CNC(C1Cc2nncn2C1)=O 3189,c1(CC)ncc(NC(=O)C(Cc2cn[nH]c2)NC(=O)Cn2ccc(C)n2)cn1 3190,c1(-n2c(C(CC(C)C)C)nc(-c3ccc(O)cc3)n2)cccc2c1CCCC2 3191,c1(CC)ncsc1C(=O)N(C)CC1(CNC(=O)CC2CCCC2C)CC1 3192,Cc1cccc2[nH]cc(CC(N3CCC=C(CNC(C4COC(C)C4)=O)C3)=O)c12 3193,c12cccc(n1)C(=O)NC2.C1(CC(=O)NCC2CCC(F)C2)(N(C)C)CCCC1 3194,C(c1cn(C)nn1)=CC(=O)NC(C(=O)N(CCCC(=O)NC)C)Cc1ccoc1 3195,C(=O)(N=S(C)(=O)c1cccc2cccnc12)c1c(N(CCN(C)C)C)nccc1 3196,C1(C(C)C)CN(C(=O)Cn2cnc(C(N)=O)n2)CCN1C(C1CCCCC1O)=O 3197,N1(C(C2C3CCCC(=O)C32)=O)CC2CCCN(C(C34CC(C3)C4)=O)C2C1 3198,c1(C(N(C(CCCC)C)C)=O)c(CNC(c2cncc(OC)c2)=O)cnn1C 3199,c1(C(N2C(C(C)(C)NC(c3cncnc3)=O)CCC2)=O)nccc2ccncc12 3200,N1(C(CCC(CC)C)=O)CCC2(CC1)CC(NC(C1CCNC(=O)C1)=O)C2 3201,Cc1cc(C(N2CC(O)CC2C(N2CCC(C)(O)CC2)=O)=O)cc(Br)c1 3202,N1(C(C(c2ccc(Cl)cc2)C)=O)CCN(C(c2nocc2C2CC2)=O)CC1CF 3203,C1(C)(CNC(CC2C(C)=NOC2=O)=O)CCN(C(=O)C(C(C)(C)C)C2CC2)CC1 3204,C#Cc1cncc(C(=O)NC(CN(C)C(C2CCS(=O)(=O)N2)=O)CC)c1 3205,n1(CC)nncc1C(=O)NCC1CC(NC(=O)C(F)(F)c2ncccn2)C1 3206,c1(C(=O)NCC2N(C(CNC(CC)=O)=O)CCC2)ccnc(N2CCCC2)n1 3207,c1(NC2C(C)C2)cc(S(=O)(=O)NCc2ccc(F)cc2)ccc1C#N 3208,C1(C(N(CC(F)F)CCOC)=O)CSCN1C(c1cc(OC)no1)=O 3209,CCC(CCC(=O)NC1CCN(CC2CC2)C1)NC(c1ccnnc1C)=O 3210,c1(C(=O)NC2CC(NC(Cn3ncn(C)c3=O)=O)C2)ccc2ncc(=O)[nH]c2c1 3211,c1(OC)cccc2c1CC(C(=O)N(C)CCN(C)C(C1CC(C#N)C1)=O)CO2 3212,C1(C(N2CCC(NC(=O)C3=CCCCO3)C(F)C2)=O)CC2CCC(C1)S2(=O)=O 3213,N1(C(C=Cc2cc(OC)c(OC)c(OC)c2)=O)CC2CCC(C1)N(C(=O)C1CC1)C2 3214,CCCCCCCCC(=O)NC12CCC(NC(=O)COCP(C)(C)=O)(CC1)C2 3215,C1(=O)C(C)(C)C(=O)N1.N1(CCCC)CCN(C(=O)COCCNC(C)=O)CC1 3216,N1(C(c2cscn2)=O)CC2(CCCCN(C(C34CC(C3)C4)=O)C2)C1 3217,N1(C(C(C=C)(F)F)=O)CCCC(CCNC(C2CC3(CSC3)C2)=O)CC1 3218,C1(OC)CN(C(=O)C=C(C)Cl)C(C)(CNC(c2ccc(C(F)F)nc2)=O)C1 3219,Cc1cc(CC(N2CCC(NC(=O)Cc3ccc(Br)s3)C2)=O)c(C)s1 3220,Cc1nc2ccc(C(N3CC(N(C)C(C4(C)CC4)=O)C3)=O)cc2s1 3221,C1(C(=O)NCCCCCN(C(COCC(C)C)=O)C)CC(S(C)(=O)=O)C1 3222,c1(C(=O)NC(C2CCCN2C(C2CCC2C(F)F)=O)C)cncc(F)c1 3223,C1(C(N2CCC(NC(c3cccc(Cl)c3F)=O)CC2)=O)CCCCCCC1 3224,Cc1cc(C(=O)NCC2CCN(C(c3ncc(Cl)cc3Cl)=O)CC2)ccc1F 3225,c1(C(=O)NCC2CC(F)(F)CN2C(C2CC3CCC2C3)=O)cn2cnnc2cn1 3226,C(=O)(C(C)CO)C(=O)NC(N)=O.C(=O)(CCO)NCCNC(=O)OCC 3227,C1(C)(CC(=O)N(C2CCN(C)C2)CC)CCN(C(c2ccccc2Cl)=O)C1 3228,C1(NC(CC(CC)OC)=O)CCC2CN(C(c3cnc4nccn4c3)=O)CC2C1 3229,C1(C(=O)NCC2(OCC)CN(C(C3(CC)CCCO3)=O)C2)CC2(C1)CC21CC1 3230,c1(NC(C(CNC(C(CCC)=CCC)=O)C)=O)c(C)[nH]c(C)cc1=O 3231,c1(OC)ncc(C=CC(N2CCC(NC(=O)Cc3ccns3)CC2)=O)cn1 3232,C(=O)(NN=c1[nH]ccnc1C1CCC1)NC(C1(OC)CCOCC1)C 3233,c1(CC)cc(C(N2CCC(c3cn(CCOC)nn3)C2)=O)nn1-c1ccccc1 3234,C1(C(=O)NC(c2ccncc2F)C)C2CCC(C2)N1C(C1CS(=O)(=O)C1)=O 3235,c1(C(N(CCCNC(=O)C(O)c2ccco2)CC)=O)c(Cl)c([N+](=O)[O-])nn1C 3236,CCCCCCN(C(=O)CC1CCCO1)CCN(C(=O)CCN1CCC1)CC 3237,N1(C(CC=C)=O)CCCC(C)(CNC(=O)CSCC)C1 3238,N1(C(COC)=O)CCOC2CCN(C(=O)C(C)OCc3ccc(C)cc3)CC12 3239,N#Cc1ccc(C(N2CCC(NC(c3ccc(-c4cc[nH]n4)cc3)=O)C2)=O)s1 3240,c1(C(N(CC(CNC(CCC(=C)Br)=O)O)C)=O)c(C)cccc1Cl 3241,N1(C(c2ccc(Br)cc2Br)=O)CC2CCN(C(c3cccc(F)c3O)=O)C2C1 3242,C=CCC(C)C(=O)NC1CCC(N(C)C(c2csc(-c3ccccc3Cl)n2)=O)C1 3243,Cc1oc(S(N)(=O)=O)cc1C(=O)NC(C1CCCN(C(C2(C)CSC2)=O)C1)C 3244,CCC(C(=O)OC)C(=O)N1CCC(CNC(=O)C(O)Cc2cn(C)cn2)C1 3245,CCCC(C(=O)NCCN(C(c1ccc(=O)n(C2CC2)c1)=O)C(C)C)C(C)C 3246,C(C)(CCCNC(=O)C(N1CCC(C)C1)=O)NC(CCN(C)CC)=O 3247,c1(C(N2CCC(C)(CO)C2)C(=O)NCCC2(C)CC2)ccc(F)c(Cl)c1Cl 3248,c1(C(=O)NC(C(C)NC(C(C)OC)=O)C)ccccc1Oc1ccncc1 3249,C1(CNC(Cc2n(C)cnc2)=O)CCCN(C(=O)CCNC(C2CCC2)=O)CC1 3250,CCCCCC(F)C(=O)NCC1CC1CNC(c1onc2c1CCCC2)=O 3251,C1(CNC(C(C)=C2CCCC2)=O)CN(C)CCN1C(=O)CNC(=O)C(F)(F)F 3252,C1(CC=C)(NC(=O)CN2CC(C)(C)C2)CCCN(C(=O)C(C)OC2COC2)C1 3253,C1(C(=O)NCCC=CCCC)CCCN1C(=O)CCn1ccc(C)n1 3254,CCC(C)(C)C(=O)C(=O)N1CCOCC(CNC(=O)CCc2ccc(F)cc2)C1 3255,N1(C(C(C(=O)OCC)F)=O)CCC(CNC(=O)Cn2nnc(=O)[nH]2)C(F)(F)C1 3256,C1(C(N2CC(O)C2)=O)(NC(=O)NCC)CCCC1.C(=O)(C(=O)N(C)C)NCC 3257,N1(C(CCCC#C)=O)CCC2CCN(C(c3cn(C)c(C)n3)=O)CC12 3258,N1(C(CCC(=C)Cl)=O)CCC(C2CCN(C(c3cc4sccc4[nH]3)=O)C2)CC1 3259,c12cc(OC)cc(c1)NC(=O)c1ccc-2cn1.c1(OCC)ncccc1OC 3260,c1(C2C(C(N3CC(OCCNC(c4cncn4C4CC4)=O)C3)=O)C2)cccnc1 3261,N1(C(C(C)COCCC2CC2)=O)CC2CN(C(=O)COc3ccccc3)CC2C1 3262,c1(SCC(=O)NCC(C)N(C(=O)CC2CCC23CCC3)C)ccccc1Cl 3263,CC(C(C)C(=O)NC1(C(O)CO)CCC1)NC(=O)CSC(F)(F)F 3264,N1(C(C2(C(C)C)CCC2)=O)CC2CCN(S(=O)(=O)c3ccccn3)C2C1 3265,CN1C(=O)CCCC1C(N1CC2CCC2(NC(=O)C(=Cc2c[nH]cn2)F)C1)=O 3266,CC(C)(C)C(O)CC(=O)N1CC2CC2(CNC(c2ccccc2C(F)(F)F)=O)C1 3267,c1(C(N2CCN(C(C3CCCN(C)C3)=O)CC2CC#N)=O)ccc(C#N)c(Cl)c1 3268,O=C(CC1CC(=O)c2ccccc21)Nc1ccc(Cl)c(S(=O)(=O)N2CCCC2)c1 3269,C(CO)(CCCCNC(c1nnc(C)s1)=O)NC(C(CC)CC1CCCC1)=O 3270,c1(NC)cccc(C(=O)NC2CN(C(C3CC3F)=O)CC2c2ccccc2F)n1 3271,N1(C(C2C(C(C)(C)C)CC2)=O)CC2CCC(C1)N2C(=O)CC(F)(F)F 3272,c1(C(N2CCC(CCC(=O)NCC(=O)NCC)C2)=O)c(C#N)ncn1C 3273,C1(C2CN(C(=O)COCc3ccccc3Cl)C2)(NC(C(C)CC2CC2)=O)CC1 3274,C=C(C)CC(C(=O)NCC(O)CN(C)C)NC(C1CN2CCC1CC2)=O 3275,N#CC1(C(N2CC3CC2CN3C(=O)C=CBr)=O)CCOCC1 3276,c1(OC)cc(NC(C2CCN(C(c3ccccc3C)=O)C2)C)ncn1 3277,C(=O)(C(CCOC)NC(C1(C)CC(C#N)C1)=O)NCCCOCCOC 3278,C(=O)(C(CCCC)N(C)C)N1CCC(O)(C(=O)NC2C(OC)CCC2)C1 3279,c1(OC2CC(OC(C)(C)C)C2)ncc(CSC(C#N)C2CC2)cn1.C1CO1 3280,N1(C(C2(CCC=C)CC2)=O)CCN(C(=O)CCn2nc(C)cc2C)CC(C)C1 3281,C1(C)(C(=O)NCC2(NC(C(N3CCC(O)CC3)C)=O)CCCC2)COCCO1 3282,c1(C(N(c2ncnc(OC)c2C)C2CNCC2F)=O)ccc(F)c(Br)c1F 3283,CC1(C)CCc2cc(C(N3CCN(C(c4cnsc4)=O)CC(O)C3)=O)ccc2O1 3284,c1(OCCCNCC(CC)(c2ccccc2)NC(C)=O)ccc(C(F)(F)F)nc1 3285,c1(CC(=O)NC2CCCC2CNC(C2(C(F)F)CCCC2)=O)c(F)cccc1Cl 3286,C1(C(N(CCC(=O)NC2C=CCCC2)CC#C)=O)CCCC(=O)CC1 3287,C1(=O)C2=NOC3(CCN(C3)N1)C2.c1(C(N2CC(C)(C)C2)=O)csc2c1CCCO2 3288,c1(C(=O)NC2(C)CCN(C(c3c(C)onc3C(F)(F)F)=O)C2)cn2c(n1)CCC2 3289,CC1Cc2cc(C(N3CCN(C(=O)CC(C)(C)C(F)(F)F)C(C)C3)=O)ccc2O1 3290,N1(C(C(CC)C(F)(F)F)=O)CCC2CN(C(c3cnc4[nH]ccnc3-4)=O)C(C)C12 3291,CC1COC(C(N2CCN(C(C3(Cl)CC34CCC4)=O)CC2)=O)CO1 3292,c1(C(N)=O)c[nH]c(C(=O)NCCOCCNC(c2nncs2)=O)c1 3293,C1(CC)COCCC1Cn1cc(CC2(C(c3nnnn3C)OC)CCCC2)nn1 3294,c1(C(=O)Nc2nc(C(C)NC(=O)OC(C)(C)C)cs2)c(C#N)ccc(Cl)c1F 3295,C1(NC(C2(C)CCCNS2(=O)=O)=O)Cc2ccccc2C1NC(=O)C=CBr 3296,Cc1[nH]c(C#N)cc1C(N1CC(c2ocnc2CNC(=O)C=CI)C1)=O 3297,N1(C(C2=CC(C)(C)C2)=O)CCC2CN(C(c3ccc4c(c3)CCOC4)=O)CC2C1 3298,C1(NC(C(c2c(C)cccc2)(C)C)=O)CC2CCC1C(NC(=O)C(O)CF)C2 3299,N1(C(CC2(C)CCCCCC2)=O)CC2(CC(NC(C3CCCS(=O)(=O)C3)=O)CO2)C1 3300,C1(C(=O)NCC[Si](C)(C)C)(CC)CN(C(=O)C(C)c2cccs2)C1 3301,Cc1cc(C(=O)NC(c2nccs2)C)c(C)n1N 3302,C1(CC(=O)NCC2C(C(=O)NCCc3onc(C)n3)C2)C(C)(C)C1(C)C 3303,c1(C(=O)NCC2CC(NC(C(c3n(C)ncc3)O)=O)C2)cc2cc(F)ccc2o1 3304,CN=c1[nH]cc(C(N2CCCC2C2(O)CN(C(c3cscc3C)=O)C2)=O)o1 3305,c1(OC(C)C)ccc(Cn2nc(-c3ccsc3)nc2CN2CCOCC2=O)cc1 3306,c1(C(=O)OCC(=O)Nc2c(C)ccc(Br)c2)cncc2c(Cl)cccc12 3307,C(=O)(N=S(C)(=O)c1cccc(F)c1)c1cn(C)c2c1cccc2 3308,Cc1cncc(CC(=O)NCC(C)(C)CN(C)C(C2NC(=O)OC2C)=O)c1 3309,C=CC(C)(CC)C(=O)NC1CC(CNC(=O)Cc2cnc(C)[nH]2)C1 3310,C(=O)(CC(C)CCC=C(C)C)N(C1CCN(C(C2CCCC(C)O2)=O)CC1)CC 3311,CN1CCOCC(NC(C2(NC(=O)C(O)CC(N)=O)CSC2)=O)C1 3312,c1(COCC)nc(NC(CNC(=O)CNC(c2cc(Cl)on2)=O)CC)cc(Cl)n1 3313,CC#CCC(C(=O)N1CCC(C(C)C#N)CC1)NC(=O)C(n1cc(C)cn1)C 3314,N1(C(c2cc(OCC)nn2C)=O)CCC(C)(CNC(c2cc(CC)no2)=O)CC1 3315,N1(C(C2CCC(C#C)CC2)=O)CCCN(C(c2cncc3sccc23)=O)C(C)C1 3316,c1(C(N2C(CNC(c3c(CC)ncs3)=O)CC(O)C2)=O)cncc(F)c1C 3317,C(=O)(CCCC(F)(F)F)NC1CC(C)(C)N(C(=O)CN2CCOCC2)C1 3318,C12(C(=O)NCC(CNC(c3ccccc3-n3cccc3)=O)F)CC1CCC2(F)F 3319,C#Cc1ccnc(C(=O)NCC(C2CC2)NC(=O)C(N2CCNC2=O)C)c1 3320,c1(CC)cc(C(=O)NC2CCC(N(C)C(c3ccnnc3)=O)C2)cc(F)c1 3321,C1(CC)CC(CC(=O)NC2CC(CNC(=O)CC(C)(F)F)C2)CCO1 3322,c1(SCC)cccc(CC(=O)NC2(CCNC(=O)CC(C)n3cccc3)CC2)c1 3323,c1(NCC(CCCC)NC(C2(CO)CCCO2)=O)cc(=O)n2cc(Cl)ccc2n1 3324,C1(CNC(CN(C)C)=O)(NC(=O)CCCC2CC2)CC2CCC1C2 3325,Cc1ccc(NC(=O)C(c2ccoc2)NC(=O)Cn2ccnn2)cc1CO 3326,N1(C(CC=CCC)=O)CC(CNC(c2ccc[n+]([O-])c2)=O)CC12CCOCC2 3327,c1(OC)csc(C(=O)NCCN(C(=O)C(n2ccnc2C)C)CC2CC2)c1 3328,n1(C(CC)C)ncc(C(=O)NC2(CCCl)CC2)c1C 3329,N1(C(c2c(OC)c(Cl)ccc2)=O)CCC2(CCN(C(=O)CN(S(C)(=O)=O)C)C2)C1 3330,C(=O)(C(C)P(C)(C)=O)NCc1c(CNC(CCNC(CC(C)C)=O)=O)ocn1 3331,N1(C(c2c(C)nsc2)=O)CC(NC(=O)CC2CC23CC3)C(c2cncn2C)C1 3332,N1(C(C2ON=C(CC)C2)=O)CC2CC1CN(C(c1cc(CO)oc1C)=O)C2 3333,N1(C(COCCCC)C)CCC2(CC1)CC(C(=O)OC)C2 3334,C1(C(=O)OC)C(C(N2CCC(NC(=O)Cc3cscn3)C2)=O)C1(F)F 3335,C(CCN=C(NCC1CN2CCN1CC2)NC(c1ccc(F)c(F)c1)C)OC 3336,C12(C(=O)NC(C)C(C)n3cccn3)CC1CN(C(=O)C(C)(C)C1CCOC1)C2 3337,c1(-c2n(C(C=C)C)nc(C(C)O)n2)cnc2cc[nH]c2c1 3338,C(=O)(C(C)(C)C(C)(C)C)N1CC(NC(c2c(C(C)C)con2)=O)C(F)C1 3339,C(=O)(C(C)S(=O)Cc1cccs1)OC(c1ccccc1)Cc1ccc(OC)cc1 3340,C12(C(=O)NC3C(C)CN(C(c4coc(Br)n4)=O)C3)CC(C)(C1)OC21CCC1 3341,c1(OCC(N2CC(N(C(CC=C)=O)CCCC)C(C)C2)=O)cccc(C)c1F 3342,c1(C(=O)NCC2C=CC(NC(=O)C=C3CCCC3)C2)cc(F)c(F)cc1Cl 3343,CC1CCN(C(=O)CCc2ccccn2)C1C(=O)N(C)Cc1nc(=O)o[nH]1 3344,C1(O)(C(C)NC(=O)CCC2CCC(O)CC2)CCN(C(c2ccon2)=O)CC1 3345,C1(C)(NC(C(CC)N(C)C)=O)CCN(C(c2cnc(O)cc2OC)=O)CC1 3346,n1(CC)ccc(C(=O)N(CCN(C)C(c2ccn(COC)n2)=O)C(C)C)n1 3347,c1(C(=O)NC(CNC(Cc2nc(CC)sc2)=O)C)c(-c2ccccc2)noc1C 3348,c1(-c2c(C(N(CCC#N)CC3CC3)=O)cncc2)cc(F)c(CO)cc1F 3349,N1(C(C2CCN(C)C2=O)=O)CCC2(CC1)CC2NC(C1(O)CC(C)(C)C1)=O 3350,C1(N(C(=O)COCCOCCO)CCO)CCCN(C(=O)CC2(O)CCCC2)C1 3351,c1(C(C(=O)N(C)CCF)NC(CC(=O)OC)=O)c(C)cccc1Br 3352,N#Cc1cc(Cl)c(Cl)cc1NC(C1CCCC12CCN(C(C1(CN)CC1)=O)C2)=O 3353,C1(c2ccccc2)(CC(N2CC(CCNC(CNC(C)=O)=O)C2)=O)CCCO1 3354,N1(C(c2c(Cl)cnc(CC)n2)=O)CCC(NC(=O)C(C2CCC2)OC)C(C)(C)C1 3355,Cc1cccc(C(N2CCC=CC2C(=O)NCCC2=CCCC2)=O)c1 3356,C1(NC(C2CCCCCC2)=O)CN(C(=O)Cn2ccc(C(F)(F)F)n2)C2CC12 3357,C1(NCc2nnn(C)n2)CCN(C(c2cccc(Cl)c2)=O)CC1(C)C 3358,C1(CC)CCC(NC(=O)CCCn2cncn2)CC1 3359,c1(C(N2CCN(C(C=C(C)C)=O)CC2c2ccncc2)=O)ccc2c(c1)CCC2 3360,c1(C(=O)NCC2(F)CCC(NC(C3(C(F)F)CC(=C)C3)=O)C2)ccc(N)c(Cl)n1 3361,C1(CCCC)CN(C(C2(Br)CC2)=O)CCN1C(c1ccsc1SC)=O 3362,c1(OC)cc(CNC(C2CCN2C(=O)C(F)OC(F)(F)F)=O)on1 3363,Cc1oc2ccccc2c1C(=O)NCCC1CC(NC(c2cc(O)nn2C)=O)C1 3364,N1(C(C2CCN(C(c3ccc4cncn4c3)=O)C2)=O)C2COCC1CC(F)C2 3365,c1(C(N2CCC(C)(CNC(C3C(C)C3(F)F)=O)C2)=O)n[nH]c2cccnc12 3366,N1(C(C2(CC)COC2)=O)CCC(NC(=O)CCOc2cccc(C)c2C)C(O)C1 3367,C(=O)(C(CNC(=O)Cc1nccn1C)C(C)(C)C)N(C)Cc1ccccn1 3368,CC(N=c1[nH]c(N(C)Cc2ccn(C3CC3)n2)nc2c1CCC2)c1csc(Br)c1 3369,c1(C(N(CCCCNC(=O)CN2CC3CC3C2)C)=O)ccc(F)c(N)c1 3370,c1(OC)cc(O)ncc1C(=O)NCCC1(O)CN(C(c2ccc(N)c(N)n2)=O)C1 3371,c1(OC(c2oc(CC)c(C)c2)=O)cc(C2CC2)cc(F)c1 3372,N1(C(C(C)SC(C)C)=O)CC2(NC(C3CCCC3)=O)CC1C2 3373,c1(C(N)=O)cccc(OCC(N2CCN(C(C3CC=CCC3)=O)CC2)=O)c1 3374,C1(C(=O)NCCC2CCC(NC(C3C(C(C)C)CCO3)=O)C2)CCC(F)(F)CC1 3375,c1(C(=O)NCC23C(CN(C(c4ncnc(C)c4C)=O)C2)C3)cc2scc(C)c2[nH]1 3376,N1(C(c2c(C)coc2)=O)CCCC(C)(C)C1C(N1CCCC(O)C1)=O 3377,c1(CC)ccnc(C(N2CC(CO)(NC(C3CN4CCC3C4)=O)C2)=O)c1 3378,C=C1CC2(C1)CC(C(=O)NCC1CCCCN(C(C3(COC)CCC3)=O)C1)C2 3379,C1(CNC(CCc2ccc(OC)cc2)=O)CC2COCC2N1C(=O)C(O)C1CC1 3380,CC1(C(=O)NCCC2CCN(C(=O)C(C3CCCCC3)F)C2)CCS(=O)(=O)CC1 3381,C1(O)(CNC(CCc2nc(C)c(C)o2)=O)CC2CCC(C1)N2C(=O)C=CBr 3382,CC1CC(CCNC(c2csc(CO)n2)=O)CCN1C(=O)Cc1cncs1 3383,Cc1c(-c2cn(CC3CC4(CC4)CN3C(=O)CCC(C)C#N)nn2)cccc1Cl 3384,C1(C(=O)NCCC2CC(NC(c3noc(CC)c3C)=O)C2)CCc2n[nH]cc2C1 3385,N#Cc1c[nH]c(C(N2CC3CC3(NC(c3cc(-c4ccccc4)cs3)=O)C2)=O)c1 3386,CC(C(=O)N1CC(CNC(c2cscn2)=O)C1)c1cc[nH]n1 3387,C12(CNC(CCc3ccc(OC)nc3)=O)CCC(NC(=O)C(C)SC)(CO1)C2 3388,c1(C(=O)NC2C(NC(C=CCN(CC)CC)=O)COC2)cccc(C#N)c1 3389,N1(C(C(CC(C)C)=O)=O)CC2C=CC1C(C(=O)N(C1(C)CC1)C)C2 3390,C=CC(C)(CCOC)C(=O)NCC1CC(NC(=O)CC(F)(F)C(F)F)C1 3391,C12(C(=O)NC3CCN(C(C4CC(C(F)F)(OC)C4)=O)C3)CCC(CC1)CC2 3392,N1(C(C(c2nc(C)sc2)=O)=O)CC(NC(c2ccc(C(F)F)nc2)=O)C(C)(C)C1 3393,N1(C(CCNS(C)(=O)=O)=O)CCC(Cn2cc(CON3CCCC3CO)nn2)CC1 3394,CN1CC=C(C(=O)NC2COCCN(C(C3(C#N)CC=CC3)=O)C2)C1 3395,c1(C(=O)NC2(CO)CN(C(=O)CC3(O)CCOC3)C2)cnn2c1OCC2 3396,C(c1cccc(Cl)c1)=C(C(N1CC(NC(C(C)(C)SC)=O)C1)=O)C 3397,CCCCC(CC)(c1nnnn1CCSCC)NC(CCO)C(C)C 3398,C1(NC(=O)CCc2cnccn2)CCN(C(c2ncccc2Br)=O)CC1CO 3399,N1(C(C(N2CCNC2=O)C)=O)CCC(C(=O)NCCCn2cnnc2)CC1 3400,N1(C(c2ccnc(C)n2)=O)CCN(C)C(C(=O)Nc2cn(C)nc2OCF)C1 3401,c1(N2CC(C)C(CNC(c3occc3Br)=O)CC2)ccc([N+](=O)[O-])cn1 3402,c1(C(N2C(CNCc3c(C)n[nH]c3)CCCC2)=O)cnc2c(c1)CCCC2 3403,CC1CC2(C(N3CC(OCCNC(C4CC(n5cccn5)C4)=O)C3)=O)CC12 3404,CC1CCCN(C(C2CCS2(=O)=O)=O)C1CNC(=O)CCN1CCOC1=O 3405,c1(C(=O)NCC2(C)C(C)CN(C(C(CCSC)O)=O)C2)cc(Cl)c(Cl)cc1N 3406,C1(CNC(CCSCCC)=O)C(C)CCCN1C(c1cc(C2(C)CC2)on1)=O 3407,C(=O)(C1c2c[nH]nc2CN1C(c1cncn1C)=O)NC(C1(O)CCC1)C 3408,c1(C(N2CC(OCC)(CNC(=O)CCc3cc(C)no3)C2)=O)cn(C)nc1CC 3409,N1(C(C2(C)CC(=C)C2)=O)CCC(CNC(c2cnn(C3CC3)c2)=O)C(O)C1 3410,C=CCCC(C)(C)C(=O)NCCC(C)(C)NC(=O)CC1CCCC(C(F)(F)F)C1 3411,N1(C(C(C)N(C(=O)CCN2CCCCC2)CC)=O)CCc2ccncc2C1 3412,CC1CCCc2ccc(NCC3CCN(C(=O)OC(C)(C)C)C3)cc21 3413,C=C(C)C(CC(=O)N1CCCC1CN(C(=O)C=Cc1ccccn1)C1CC1)OCC 3414,C1(NC(C2(CC=C)CC=CC2)=O)COCCC1NC(=O)CCN1CCOCC1 3415,c1(-c2n(-c3c(C)cccc3)nc(-c3cccnc3)n2)c(C)cc(C)c(CO)c1C 3416,c1(C(N2CCCC2c2cn(C3CCC3)nn2)=O)cnc(CC2CCOC2)s1 3417,C(=O)(C1=CC2CCCC12)N(C1CCN(C(c2ccc3nncn3c2)=O)C1)CC 3418,C(=O)(CCCCC(=O)OC)N1CCN(C(COCCC=C)=O)CC1C(C)(C)C 3419,CCC(F)(F)C(=O)NCC1CCCC1NC(=O)Cc1cn(C2CC2)cn1 3420,CC1(CCC(=O)Nc2cnsc2)CCCN1C(c1ccc(Cl)s1)=O 3421,C1(N(C(=O)Cc2csc(Cl)n2)C)CN(C(=O)C#CC2CC2)CC12CC2 3422,C1(CNC(CC(=C=C)C)=O)CN(C(=O)C(CCC)NC(C)=O)CC12CC2 3423,c1(NC(N2CC(C(C)N(C)C)C2)=O)cc(F)ccc1N1CCN(C)CC1 3424,N1(C(C(C)C(F)F)=O)CC(CC(=O)NC2CCN(C(N)=O)CC2)C2(CC2)C1 3425,N1(CC(=O)NC2C3CN(C(c4n(C)ncc4Cl)=O)CC2C3)C(=O)NC(C)(C)C1=O 3426,C1(C(N2C(C(=O)NC3(CC=C)CC=CC3)CCCC2)=O)C2CCCC(=O)C12 3427,Cc1ncc(NC(C2C3CCN(C(=O)C(C)SC(C)C)CC23)=O)c(C)n1 3428,CCCC(CNC(c1cccn1C)=O)C(=O)N(CC)CC1CCCO1 3429,c1(N(c2cnn(C)c2)C)nnc(-c2cnsn2)n1C 3430,C1(CC(=O)NCCn2ncc(CC)c2)CCN(C(c2cnc(NC)cn2)=O)CC1 3431,N1(C(C(c2ccc(Br)cc2)C)=O)CCCC12CCN(C(=O)CCCC#N)C2 3432,Cc1cc(=O)ccn1CC(=O)NCCCN(C)C(c1coc(C(F)(F)F)n1)=O 3433,C12(C(=O)NC3(CC(=O)OCC)CC3)CC(CN(C(=O)CC3CC(C)=NO3)C1)C2 3434,c1(OCCC)nc(C)ccc1C(N1CC2(C1)CN(C(c1ncc(CC)[nH]1)=O)C2)=O 3435,Cc1cc(S(=O)(=O)C(C2CC2)OC(C)(C)C)c(C)cc1-c1cccc(N(C)C)c1 3436,C=CCC(CC(C)C)C(=O)NC1CC1NC(c1c(C)nn2ccccc12)=O 3437,C1(NC(Cc2cc(OC)no2)=O)C2CN(C(C3CC(C)OC3C)=O)CC12 3438,N1(C(C2C(C(C)C)C2)=O)CCC(OCCCNC(C2(CC#N)COC2)=O)CC1 3439,c1(C(=O)NC(CNC(c2c(CC)cno2)=O)CCOC)c(Cl)n[nH]c1CC 3440,OC1CCC2(CC1)CCN2c1nnc(-c2coc(Br)n2)o1 3441,c1(OC)ccc(O)cc1C(N1CC2CC1CC2NC(c1ncc[nH]1)=O)=O 3442,N1(C(c2c(C)nc(CC)o2)=O)CCN(C(=O)COCC2CCOC2)C(C(F)F)C1 3443,C(=O)(C1=CCC(C)(C)CC1)N(C1CCN(C(=O)C(O)C(C)SC)CC1)CC 3444,Cc1ncc(NC(C2CC(O)CN2C(C2C3(CC3)C23CC3)=O)=O)cc1C#N 3445,Cc1cc(F)ccc1C(N1CCC(N(CCO)C(C2OCC2(C)C)=O)C1)=O 3446,N1(C(c2cc(C)n(C)c2)=O)CC2(C=C(C(=O)N(C3CCCCC3(C)C)C)CO2)C1 3447,C(CC(C)C)(C(=O)NC1CCN(C(=O)C(F)C(C)C)C1(C)C)OC 3448,Cc1c(F)cc(CNc2cccc(C(=O)Nc3c(F)cc(Cl)cc3Br)c2)cc1Br 3449,c1(C(=O)NC2C3CN(C(C4(C#N)CC45CCC5)=O)C(C3)C2)ccc2c(c1)OCC2 3450,C(CO)(CCCCNC(=O)Cc1csc(C(C)(C)C)n1)NC(C1(F)C(C)C1)=O 3451,CCCCCCCC(=O)N1CCCC(C(C)NC(c2cccc(Cl)c2F)=O)C1 3452,C1(C(=O)NCCCN(C(=O)CCn2cnccc2=O)C)CN2CCN1CC2 3453,C1(C(=O)NCC=CC(=O)N(CC(COCC)O)C)CCC(C)O1 3454,C1(NC(CC2(COC)CCCC2)=O)(CO)CCN(C(=O)CC2CC(C)(C)CO2)C1 3455,c1(C(=O)NC2CN(C(C(C)(C)N3CCOCC3)=O)C2)ccc2cc[nH]c2c1 3456,c1(C(N2CCC(NC(CC3=NNC(=O)C3)=O)C(F)C2)=O)cc(=O)n2nccc2[nH]1 3457,c1(C(=O)NC(C(C)(C)NC(C=C(C)C)=O)C)cc2[nH]nc(C)c2cn1 3458,N1(C(CC=CC)=O)CCN(C(C2CCCN(C)C2)=O)C(c2cn[nH]c2)C1 3459,CCCC(C(=O)NCCC1CN(C(c2cccnc2-n2ccnc2)=O)C1)OC 3460,C1(NC(C2C(NC(C(C)S(N)(=O)=O)=O)CC2)=O)CCC2(CCC2)CC1 3461,c1(SCC)ccc(C(N2CCC(COC)(NC(=O)C(C)c3cc[nH]n3)C2)=O)cc1 3462,C(=O)(C(CCOCC)NC(=O)COCCCC)NCC(=C)F 3463,CC1(CNC(C2C3(CC3)C23CC3)=O)CCN(C(=O)C=Cc2cnc[nH]2)CC1 3464,C=C(C)C(C)(O)C(=O)NCCOC1CCN(C(c2cccc(SC)c2[N+](=O)[O-])=O)C1 3465,Cc1nn(C(C)C)cc1C(N1CCCC(NC(C23CCC(CC2)O3)=O)C1)=O 3466,C(CNC(C1CCN(CC(C)C)CC1)=O)(C(C)C(C)C)NC(c1cc(C)ns1)=O 3467,C1(NC(C(CC#C)O)=O)CN(C(=O)C=C2CCC2)CCC1(C)C 3468,C1(CC)CN(C(C2C(C)(C)C2(C)C)=O)CCN1C(c1cc(OC)ccn1)=O 3469,C1(NC(C(CN(C)C)NC(c2c(CC)ncnc2)=O)=O)CCc2n[nH]cc2C1 3470,N1(C(c2cc(C)sc2)=O)CC(C)OC2(CCN(C(c3ncccc3F)=O)CC2)C1 3471,N1(C(C(C(=O)NC)(C)C)=O)CCC2(CCN(C(c3coc(C(F)F)n3)=O)C2)C1 3472,C1(CCC(C)(C)NC(C2C(=C)C2)=O)CCCCN1C(=O)CC1CCOCC1 3473,c1(NCC2CCCN(C(CCC(C)OC)=O)C2)c(C(C)=O)cc([N+](=O)[O-])cc1Cl 3474,Cc1nc(C)c(C(=O)NCC2(CNC(=O)CCC(=O)N(C)C)CCOCC2)[nH]1 3475,N1(CC=C(C)C)CCN(C(=O)C(Cc2ccoc2)NC(C2CNC(=O)N2)=O)CC1 3476,CN1CCCCCC1C(=O)NC1CC(CO)N(C(=O)C2=COCC2)C1 3477,C1(NC(c2ccnc(C)n2)=O)COC2(CCN(C(c3cccc(=O)o3)=O)C2)C1 3478,n1(CN(C2C(C)C2)C)c(N2CCOCC2)nnc1-c1cnn(-c2ccccn2)c1 3479,c1(OC)cccc(COCC(=O)NC2CC(CNC(=O)COC(F)F)CC2O)c1 3480,c1(CN2C(CNC(c3cccnc3F)=O)CC(F)C2)cnc(O)nc1O 3481,N1(C(=O)NC)Cc2ccc(CNC(N)=O)nc2C1.C1(=O)CC(c2ccccc2)N1 3482,CC1CN(C(N2CCC(N3CCCC3)C2)=O)CC1CS(N)(=O)=O 3483,CC1CN(C(=O)CCc2ccc(O)nn2)CCCN1C(c1ccc(F)cc1Cl)=O 3484,N1(C(=O)Cc2ccco2)CCOC(CC(N2CCCOCC2)=O)C1 3485,c1(C(=O)NC(CCOC)CNC(=O)C(C)CSC(F)(F)F)cnc(C#N)s1 3486,N1(C(C2(c3c(C)cccc3)CCCC2)=O)CC2(CCN(C(=O)CC(C)F)CC2)C1 3487,C1(C(N2CCCC2CN(C)C(c2nscc2Br)=O)=O)(OC)CCSC1 3488,S(=O)(=O)(c1cc(C(N2CCC3(CC2)CC(CNC(=O)C2CC2)C3)=O)n(C)c1)NC 3489,Cc1nn(C)c(C(=O)NCc2cc(O)nc(CNC(=O)C(C)O)n2)c1Cl 3490,C(=O)(C(C)(C)CC(C)C)NC1(C(=O)OC)CCN(C(C2CC2C2CCCC2)=O)C1 3491,C1(C(=O)NCc2cc(CO)on2)(COC)CN(C(=O)CCc2cnc[nH]2)C1 3492,C1(NC(C2ON=C(C)C2)=O)CCC2(CC1)CC2NC(c1cncc(O)c1)=O 3493,c1(C(=O)NCCCCC2CN(CCn3ncnc3CO)C2)cnc2c[nH]nc2c1 3494,C1(C#CC(=O)NC2CCC(CNC(c3csc(C(C)=O)n3)=O)C2)(CC)CC1 3495,c1(C(C)C)noc(CCCC(=O)N2CCC(CN(C(=O)Cc3cnns3)C)C2)n1 3496,CN1CC=C(C(=O)NC2CCC(NC(=O)C(CCO)N(C)C)CC2)C1 3497,N1(C(CCCC(=O)NC)=O)CCN(C(C2(CCOC)CCC2)=O)CC12CCC2 3498,C(C(CCC)C(=O)N1CCCC1CC(=O)OC)NC(COC1(C#C)COC1)=O 3499,N1(C(C2C(NC(C3CCCC3F)=O)CCOC2)=O)C2C=CCC1CCC2 3500,C(=O)(CS(C)(=O)=O)N1C(C(=O)NC(C=C)(C)CC)CC1 3501,Cc1cc(C(N2CCCC2CCCNC(=O)CCc2cnc[nH]2)=O)cc(C)c1F 3502,c1(CC(=O)NC2CC(NC(c3ccc(F)cc3O)=O)C2)cc(F)cc(Cl)c1 3503,C1(C(N2C(CN(C(=O)C=C3CCC3)C3CC3)CCC2)=O)CC2C=CC1C21CC1 3504,c1(OC(CC)C)cc(NCC2(O)CCN(C(C3CCCC3C)=O)CC2)nc(C)n1 3505,c1(C(N2CC(NC(CSCC)=O)C(CO)CC2)=O)cc2c(C)sc(C)c2s1 3506,Cc1cnc(CCNC(C2CCN(C(=O)C(O)CC3CCCC3)C2C)=O)nc1 3507,CC1OC(=O)NC1C(=O)NCC#CC(=O)NCC#CCCO 3508,Cc1ccc(-c2nc(CC(C3CCCO3)N(C)C)n(-c3ccccc3)n2)cc1 3509,c1(C(=O)NC2CC(OC)C(OC)C2)ccc(CSC)cc1F 3510,N1(C(c2cc(C)c(O)cc2)=O)CC(C)(CNC(C2CCC(=O)NC2)=O)CC1(C)C 3511,CC(C)CC(c1nc[nH]n1)N(c1ccccc1)C(=O)C(n1cc(C2CCC2)nn1)C 3512,N(C1CCc2ccccc21)(CC(=O)OC)C(=O)COCCNC(=O)N(CC)CC.CCC 3513,C1(C(C)C)C(NC(c2cc(Cl)ccn2)=O)CCN1C(C1CC1c1ccn(C)c1)=O 3514,CC1CN(C(=O)CSCCC#N)CCC1CNC(=O)Cn1ccccc1=O 3515,N1(C(C2(CC)COC2)=O)CCC2(CC(NC(c3ccnc(Cl)c3OC)=O)CO2)C1 3516,N1(C(c2ccc(C)c(Cl)c2)C(=O)NC(C)(C)C)CCOCC2(COCCN2C)C1 3517,c1(C(N2CC(O)CC(NC(C=CSC)=O)C2)=O)cc2cc(Br)ccc2o1 3518,c1(C(=O)NC2(C(=O)NCC(C)(C)C#N)CC2(C)C)ccc(C#N)cc1 3519,N1(C(C(CC)NC(N)=O)=O)CC2(CC(NC(c3cnc(C)s3)=O)CO2)C1 3520,c1(CC)ccc(C(N2CC(CNc3ncc(Br)c(C)n3)CC2C)=O)cc1F 3521,C(CC1=CCN(Cc2ncsc2Br)CC1)NC(C1CCCC(F)C1)=O 3522,c1(OC)ncnc(OC)c1CNC(C1N(Cc2cc(CO)ccc2F)CCOC1)=O 3523,c1(C(=O)NCC2C(C)CN(C(C34CC5CC3C4C5)=O)CC2)ccn2ccnc2c1 3524,N1(C(CSc2ccc(OCC)cc2)=O)CC(C(=O)O)c2ccccc21 3525,N1(C(C(CCC)=CCC)=O)CCCCC(NC(=O)C(C)N2CC(C)C2)C1 3526,C(CCCCCCC(=O)NCCCCCCN(C)C)NC(C(CCC)OCC)=O 3527,N1(C(C(C(C)C)NC(N)=O)=O)CC(NC(c2coc(C3CC3)n2)=O)C2CC2C1 3528,c1(CC(=O)N(CC(C)CNC(=O)C(C)OCC2CC2)C)cc(Cl)ccc1Cl 3529,C#Cc1cccc(C(=O)NCC2CCCCC2NC(C2CCSCC2)=O)c1C 3530,c1(C(=O)NC2CC(C)CN(C(C3(O)CCOC3)=O)C2)ccc(S(N)(=O)=O)c(F)c1 3531,Cc1cc(C(N2CC3CC(NC(=O)CCCc4ccccn4)C3C2)=O)cc(O)n1 3532,c1(CN2CCC(CC(N3CCC3CNCCCl)=O)C2)nc(Cl)ccc1F 3533,C1(C(=O)NCc2nn[nH]n2)(COC)C=CCN1C(c1cc(C)sn1)=O 3534,N1(C(C(C)(C)CF)=O)CCC(CNC(=O)C(c2ccc(F)cn2)(F)F)C(F)(F)C1 3535,C1(C(=O)NCCC2(O)CN(C(c3nccc(C)c3)=O)C2)CCCS(=O)(=O)C1 3536,Cc1nc2n(n1)CC(C(=O)N(CC(c1ccccc1)C1CCC1)C)CC2 3537,N1(C(CCN(C(C(C)NC(CC)=O)=O)CCCO)=O)CCN(C)C(C(C)C)C1 3538,C(=O)(C(CCCC=C)NC(=O)C=CCCC(C)C)N1C(CCC#C)CCC1 3539,c1(C(N2CC(SC)C(NC(C3C(C)C3C)=O)C2)=O)cc(C#N)ccc1Cl 3540,c1(C(=O)NCC2C(CNC(CC=C)=O)C2)c(C)nn(-c2ccc(Cl)cc2)c1C 3541,CCC(CC(=O)N1CCC(CC)(NC(c2c[nH]cc(C)c2=O)=O)CC1)C(C)C 3542,c1(C(N(C)CC2N(C(C(C3CCOC3)OC)=O)CCCC2)=O)cc(C#N)n(C)n1 3543,C1(NC(C(c2ccc(OC)cc2C)C)=O)CN(C(=O)C(N)=O)C2(CCCC2)C1 3544,N(C(=NCCc1cc(Cl)ccc1Cl)NC1CC1C1CC1)C(C)C 3545,c1(C(C)NCC=C(Cl)Cl)ccc(C(C)(C)C)cc1 3546,C1(CC(=O)NCCOC2CCN(C(c3cccc(CF)c3)=O)C2)CCCS1(=O)=O 3547,C(=O)(C1=CCCOCC1)NCC(C(N1CC[Si](C)(C)C1)=O)CC1CC1 3548,Cc1cc(C(=O)NC2CC(CNC(c3[nH]cnc3C)=O)CC2O)nnc1O 3549,C1(C(=O)Nc2cnn(C3CCNC3=O)c2)CNCC2(CCC2)O1 3550,C1(N(C(C)C)C(=O)NCC(C2CCCO2)O)CCN(C)CC1 3551,C#CCC(C(=O)N1CCC(CC(=O)Nc2ccccc2OCC)C1)C1CC1 3552,Cc1cc(C(=O)NC2CCN(C(c3cn(C)nn3)=O)CC2C)ccc1Cl 3553,C(CC(C)C)(C(=O)N1CC(CNC(c2c3c(nn2C)CCC3)=O)C(C)(C)C1)OC 3554,S(=O)(=O)(c1cccc(Oc2ccccc2)n1)N(C(CCC)C(=O)O)C 3555,c1(C(=O)OC)cc(NC(=O)NC(c2cccc(OC(F)F)c2)C)ccc1F 3556,N1(C(C2CN(C(=O)NC)C2)=O)CC(C2(NC(c3nc(C4CC4)oc3C)=O)CC2)C1 3557,C(C(=O)N1CCN(C)C(C(N2CCC2CC2CCCC2)=O)C1)(C(C)(C)C)N(C)C 3558,N1(C(C(C=C)O)=O)CCC2(CCC(NC(c3cc(C)c4[nH]nnc4c3)=O)CC2)C1 3559,n1(CC#C)cccc1C(=O)NC1(C(=O)NCC2CN(C(C)C)C2)CCSC1 3560,N1(C(c2ccc(Cl)c(C(F)F)c2)=O)CCc2ccc(Br)cc2CC1 3561,c1(CNC2(CO)CC(F)(F)C2)cn2ccccc2n1 3562,c1(C(N2C(CCC(=O)NC(CC=C)C3CC3)CCC2)=O)ccc([N+](=O)[O-])[nH]1 3563,C(=O)(C1=NN2CCCN=C2N1)NC(CNC(=O)C=CC=C(Cl)Cl)C1CCC1 3564,C1(CN(C(Cc2cn(CC)nc2)=O)C)C2CN(C(C3CCCC3O)=O)CC12 3565,c1(OC)ccc2c(C)c(C(=O)NC3CCC4(CC3)CC4)[nH]c2c1 3566,c1(C(N(CC(CN(C(=O)Cc2cnoc2)C)O)C)=O)ccn(CCF)n1 3567,C1(F)(CNC(c2nc(CC)oc2C)=O)CCCN(C(c2ccon2)=O)C1 3568,N1(C(=O)Cn2ccc(C(F)(F)F)n2)CCCC2CCN(C(=O)C3=COCC3)CC12 3569,C=Cn1nncc1C(=O)NC1(CN2CCN(C(=O)C(C)O)CC2)CC1 3570,c1(CCCSC)cn(C(C)CNC(C2CC2(C)C)=O)nn1 3571,S(=O)(=O)(c1c[nH]ccc1=NC(CF)CF)NCc1cc(C)no1 3572,Cc1ccsc1CCCC(=O)NCCOCCNC(=O)C(C)C1(O)CCC1 3573,c1(C(=O)NCCC(=C)CNC(c2cc(C)nn2C)=O)c(Cl)ccc(Cl)c1OC 3574,C1(CNC(CCCCC=C)=O)CN(C(=O)C(F)(F)C(O)CC)CCC1(C)C 3575,C(=O)(C(C)(CC)CCC)N1CC(C(C(N2CCCC(OCCC)C2)=O)O)C1 3576,CCS(=O)(=O)CC(=O)NC(C)C(C)NC(c1ccoc1C(F)(F)F)=O 3577,C(=O)(C(CN(C)C)c1ccccc1)NCCN(C(C1CCCCC1)=O)CC 3578,C1(C(N(CC(=O)NC(C)C)C)=O)(CO)CCN(C(c2cnn(C)c2N)=O)C1 3579,C1(C(=O)NCCC(C)NC(c2nc(COC)sc2)=O)COCCN1CC(F)(F)F 3580,c1(C(=O)NC2C(CNC(C3(C#C)CC3)=O)C2)ccc2c(c1)CCN2S(C)(=O)=O 3581,N1(C(CC(C)(F)F)=O)CC2(CCC(NC(=O)CC3NC(=O)NC3=O)CC2)C1 3582,C1(C)(CNC(CNC(=O)OC(C)(C)C)C2CC2)CC2(C1)CC(F)(F)C2 3583,C1(C(=O)NCCCNC(C(C(C)(C)C)O)=O)CC(O)c2ccccc2O1 3584,C(=O)(C1CCc2nccn21)NCC(=O)NCc1c(C)nsc1 3585,CC1=C(C(=O)N(C2CCCC(N(C)C(C)C)C2)C)CCS1(=O)=O 3586,N1(C(C2CCC(NC(C3(SC)CC(=O)C3)=O)CC2)=O)CCN2C(=O)OCC2C1 3587,c1(C(N2CCN(C(Cc3scc(C)c3)=O)CC2C)=O)nn(C)c2c1CCC2 3588,c1(CC)nc(O)c(C(=O)NCC(C)NC(c2oc(Br)cc2C)=O)cc1C 3589,C(CC(F)(F)Cn1cc(CCC(C)O)nn1)NC(c1c(CC)occ1)=O 3590,C1(NC(CC2(OC)CC2)=O)CCN(C(C2(OC(C)=O)COC2)=O)C1.C(C)(C)C 3591,CCC(CN(C)C)CC(=O)NC1CN(C(=O)C(C)NC(=O)CC2C=CCC2)C1 3592,C(=O)(CC(C)(C)NC(C1C=CCS1)=O)N(C)C 3593,C1(CNC(CCCc2ncc(C)o2)=O)CCCN(C(c2sc(C)nc2C)=O)CC1 3594,Cc1cnc(NC(CNC(C2CC23CCOC3)=O)C2CCC2)nc1O 3595,C#CCCCCC(=O)NCC(C)(O)CNC(c1ccc(C(=O)C2CC2)cc1)=O 3596,C1(NC(c2ccc(CNC(CC(C)O)=O)cn2)=O)CCCN(C)C1C 3597,c1(C(=O)NC2C(NC(c3c(N)nc(Cl)cc3)=O)COC2)cnn2c(=O)cc[nH]c12 3598,C(=O)(CC(C)CC(C)(C)C)NCC1N(C(C(C)C)=O)CC1 3599,C(CCC)(C(O)C(=O)N1CC=CC1CF)NC(C(C)OCC#C)=O 3600,N1(C(c2c(OC)csc2)=O)CCCN(C(c2cn(CC(F)F)cn2)=O)C(CO)C1 3601,c1(C(=O)NCCC(CNC(=O)C=Cc2ccccc2)O)cccc2ccnn12 3602,C(CC(=O)NC1CC1C(N1CCC1C)=O)OC 3603,c1(CNC(c2sc(C(=O)NC3(C)CN(CC)C3)c(C)c2)=O)ccc(C)c(C)c1 3604,N1(C(C(C(CC)(C)C)O)=O)C2CCCC1CN(C(=O)C(CO)OC)C2 3605,N1(C(CCN(C(=O)CC2CCOC2=O)CC#C)=O)CCC2(CC1)CC2C#N 3606,C1(CNC(c2ccc(OC)cn2)=O)CC2CN(C(c3cc(C)nc(C)c3)=O)CC12 3607,C(=O)(C1=C2CCN=C2NC=C1)N1CCC(N(C(=O)CS(C)(=O)=O)C)CC1 3608,C(N=c1nc(N2CCC3(CCCN(C)C3)C2)c2sccc2[nH]1)C1(C)ON=C(C)C1 3609,c1(OCC)ccc(Cl)nc1C(=O)NC1CCN(C(=O)CCCOCCOCC)C1 3610,CC1CC(c2ccccc2)CC(C)N1CC(C)(C)CO 3611,Cc1ccc(C(=O)NC2CCC(C)N(C(C3CC4CCC3CC4)=O)C2)cc1CO 3612,c1(CC)cccc(C(=O)NC2CC2NC(=O)COc2ccc(C)cc2)c1C 3613,N1(C(=O)C(=O)CC(c2ccccc2)N)CCC2(CCNC2=O)C1.c1(O)ccccc1 3614,C1(CC(=O)N(CCC(N)=O)C)CN(C(c2cc(O)cc(=O)o2)=O)C(C)(C)C1 3615,N1(C(COCCC)=O)CCC(C(=O)NCc2cn(C3CC3)nn2)C1C 3616,c1(NC(C=CCNC(c2cc(C(C)=O)on2)=O)=O)cnc(O)cc1C 3617,c1(C(=O)NC(C)C(C)(C)NC(C2CCC(F)(F)C2)=O)cccc[n+]1[O-] 3618,c1(C(=O)NC(C2CN(C(=O)COC3(C)CCCC3)C2)C)ccc(C2CC2)cn1 3619,CN1CCC(C(=O)NCC23CC(CNC(=O)CC(F)(F)F)(CO2)C3)CC1=O 3620,c1(SC)ccc(C)c(C(N2CCOCC2CNC(c2ccc(C)c(C)c2)=O)=O)c1 3621,C(C(C)(O)CC(=O)N(C1CN(C(c2c[nH]nc2C)=O)CC1(C)C)C)OC 3622,c1(CC(=O)OC)ccc(C2CNC2)cc1.C1C(C)C(=O)NC(=O)C(=O)N1 3623,C1(C)(C(N(C(CNC(=O)CCC2CCCOC2)C2CC2)C)=O)CCCO1 3624,C(=O)(C(C)(C)C(C)(C)O)N1C(CN(C(c2cccc(CSC)c2)=O)C)CCC1 3625,c1(N2CC3CC4C(O)C2C3C4)nc(C2CC2)nc2c1CCC2 3626,c1(C(N(C2CCCCC2)CCNC(=O)Cc2ccoc2)=O)nsnc1O 3627,Cc1nc(NC(C2(C(F)(F)F)CCN(C(C)C)C2)=O)ccc1[N+](=O)[O-] 3628,C(CC(CC)C(=O)NC1C=CCC(C(=O)N(CCN2CCOCC2)CC)C1)=CC 3629,C1(CNC(c2c(CC)scc2)=O)CCC2CN(C(C3CN(C)C(=O)N3)=O)CC12 3630,C(=O)(C(CNC(c1cc(CO)n(C)n1)=O)C(C)(C)C)N(CCn1ncc(C)c1)C 3631,N1(C(CCCC(C)n2cc(-c3cnc(C(=O)OC)s3)nn2)=O)CC2(CCCCC2)CC1C 3632,C(=O)(CN=c1cc[nH]cc1)N1CCC=C(CNC(C2CCOC2)=O)C1 3633,C=CC(O)(C(=O)NC1CCCCC1NC(=O)CSc1ccccc1)C(F)(F)F 3634,c1(CC)cc(C)c(C(=O)NC2CC2CNC(=O)CNc2ccc(NC)cc2)o1 3635,C1(C(=O)NC(C)C)CC(NC(C2CC(C)(C)CO2)=O)C(O)C1 3636,C1(CCCNC(C(F)=CCC)=O)CN(C(c2ccnc(OC)n2)=O)CCO1 3637,n1(CC(=O)N(CCCCCNC(C2CC2Cl)=O)C)ccc([N+](=O)[O-])n1 3638,CCC(CNC(C1CN(C(=O)CCC(C)(C)C)CCN1C)=O)CC(C)C 3639,C(CC(=O)NCCC(O)C1CC1)(C(F)(F)F)NC(C1(COC)CCCC1)=O 3640,N1(C(=O)CC(F)(F)CCc2ccccc2)CCC2(CC1)CC(F)CO2 3641,C1(NC(C2N(C)CCCC2)=O)CCN(C(=O)CNc2cnn(C)c2)CCC1CO 3642,C=CCC(CC(C)C)C(=O)N(C(C)CCNC(c1nccc2ccccc12)=O)C 3643,N1(C(C(C)CSC(F)(F)F)=O)CC2CCN(C(c3nnn4c3CSCC4)=O)CC12 3644,c1(C(=O)NC2C(CNC(Cc3nc(C)sc3C)=O)CCCC2)cccc(Cl)c1N 3645,C1(NC(c2cc(CCC)[nH]n2)=O)CC(O)CN(C(=O)Cn2cc(F)ccc2=O)C1 3646,C(CC(O)C(F)(F)F)NC(C(CC=CC)NC(=O)CC1CCOC1=O)=O 3647,C(=O)(C1=COCCC1)NCC(CC(C)C)NC(=O)C(c1cncn1C)O 3648,N1(C(C2CCCC(OC)C2)=O)CCC2(CC1)CCN(C(C1CC1C)=O)CC2 3649,CCC(C)C(C(=O)NCCCCC(=O)NCC(C)CCOC)N(C)C 3650,N1(c2ncc(C(=O)OC)c(C)c2)CC2CC(NC(=O)CCC(C)(C)O)CC1C2 3651,c1(C(=O)NC(CNC(C(C(C)C)n2cccc2)=O)CO)cn2cnnc2cn1 3652,c1(CC(C)C(=O)NC(C)(C)C)ccc(F)cc1.c12ccc(o1)COCCNC2=O 3653,N1(C(C2(COC)CCCOC2)=O)CCC2(CC1)CC2CNC(=O)CC(C)(F)F 3654,C(=O)(CCN(OC)C(=O)c1ccc(C#N)[nH]1)N1C(C)CC1 3655,N1(C(Cc2ccc(C)cc2)=O)CCCC(C)C1CNC(=O)C=CC1CCOCC1 3656,c1(C(=O)NCC2CC2NC(=O)C(O)Cc2ccc(Cl)cc2)nccc2[nH]ccc12 3657,C1(C(=O)Nc2cn(CCOC)nc2)CCC(C)(C)N(C(c2csc(O)n2)=O)C1 3658,CC1CC2(CCO1)CC2C(=O)NCC1(CNC(c2coc3c2CCCC3)=O)CC1 3659,c1(C(=O)NCC2(OC)CN(C(c3ccnc(OC)n3)=O)C2)c(C)cnnc1O 3660,N1(C(C(C2CC=CCC2)NC(C(CC(N)=O)O)=O)=O)CCC(C2CCC2)CC1 3661,N1(C(COC)C)CC(NC(c2ccc(C)nn2)=O)C(C)(C)C1 3662,N1(CC)CC2CN(C(=O)C(CC)NC(c3ccc(F)cn3)=O)CC2C1 3663,Cc1c[nH]c(C(N2CCN(C(=O)CCCc3cccs3)C(C)C2)=O)cc1=O 3664,C(c1cscn1)=CC(=O)N(C1CCN(C(c2sccc2CC#N)=O)C1)CCC 3665,c1(CN(C(C=C(COC)C)=O)C2(NC(=O)OC(C)(C)C)CC2)ccnc(C)n1 3666,c1(NCCNC(C2(N(C)C)CCCC2)=O)ncnc2ccccc12 3667,c1(C(=O)NCC#CCNC(=O)C2=CCCS2)coc2c(Cl)cccc12 3668,Cc1nc2cccc(C(=O)NC3CC(NC(c4cc5sc(C)c(C)c5[nH]4)=O)C3)n2n1 3669,CCC(C)C(O)C(C)C(=O)NCC(C)(C)C(N1CCCC(F)(F)C1)=O 3670,N1(C(C2(SCC)CC2)=O)CCCC(CC)(NC(c2cc(C(C)=O)oc2C)=O)C1 3671,c1(C(N(CC(C)(C)CNC(=O)Cc2nncn2C)C)=O)cnc2c(c1)ncn2C 3672,N1(C(C2CC(CC)C2)=O)CCN(C(c2ccc(Cl)nc2N)=O)C2CC12 3673,C1(C(N(C(CNC(c2cnc(CC)s2)=O)C)C)=O)(OC)CCC(F)(F)CC1 3674,Cc1cc(C)c(C(=O)NC(C)(C)C(C)NC(c2cncc3ccsc23)=O)cc1C 3675,C1(NC(c2n(CC)ccc2)=O)CN(C(=O)C=CC2CCCO2)CC2(CCC2)C1 3676,N1(C(C)C)CCCC1C(=O)NCCC(C)(C)NC(=O)C(C)CC1CCCCC1 3677,c1(OCCC(=O)NC2CCC2NC(=O)C(=O)NC2CC2)ccc(Br)cc1 3678,N1(C(C(CC)C(C)C)=O)CC2CCCC(NC(C3CCCS(=O)(=O)C3)=O)C2C1 3679,c1(C(=O)NCC(COC)NC(c2c[nH]nc2C)=O)ccc2n[nH]cc2c1Cl 3680,n1(CC)nccc1C=CC(N1CCCC1CN(C)C(C1COC(=O)N1C)=O)=O 3681,c1(C(=O)NCC2CC(OC)CN2C(=O)C(C)C2CCCC2)c(Cl)c(C)nn1C 3682,N1(C(=O)OC(C)(C)C)CCC(CC(c2ccc(O)cc2)O)CC1 3683,C(=O)(C(O)CCS(C)=O)NC1(CNC(C(CN(C)C)(C)C)=O)CCC1 3684,N1(C(C(C)OCC2CCCO2)=O)CCN(C(C2CCCS2(=O)=O)=O)CC1 3685,c1(C(N(C2CCCC(NC(c3cc(C)oc3C)=O)C2)C)=O)cnc2n1CCCC2 3686,N1(C(C(CSC)OC)=O)CCN(C(c2cnnc(O)c2)=O)C(C)C1 3687,Cc1nn(C2CC2)cc1C(=O)NC(CNC(=O)CC(O)c1ccccc1)CO 3688,C(=O)(C(CNC(=O)C=Cc1ccncn1)CC1CCCC1)NC1C(CC)CCC1 3689,N1(C(C2(CC)CC=CC2)C(=O)NCC2CCCO2)CCC(C)(CCO)C1 3690,Cc1ncccc1C(=O)NC1CC1C(N1CCC(Cc2ccc(Br)cc2)C1)=O 3691,C(=O)(C#CC1(C)CCCO1)N1C(C)(C(NOCCCOC)=O)CC(O)C1 3692,CC1(C)OC(=O)CC1C(N1CCCC(C(=O)Nc2ccc(F)cc2)C1)=O 3693,N1(C(CC)=O)CCC(C)(C(=O)Nc2cnc(C(F)(F)F)nc2)C1 3694,C1(NC(C(CC)(C)O)=O)CN(C(=O)CCn2ccnc2C)CC(C)(C)C1 3695,N1(C(C(CC)n2ccnc2)=O)CC2(CNC(c3ccc(COC)o3)=O)CC1CO2 3696,n1(CCNC(CC(C(C)C)c2ccc(F)c(F)c2)=O)cnc2c1CCCC2 3697,C(=O)(C(C(=O)N(C1CCN(C(=O)C(c2cccc(C)c2)(C)C)C1)C)OC)OCC 3698,N1(C(CCc2cnc(C)o2)=O)CCN(C(C2CCCC2C(F)(F)F)=O)CC1CO 3699,C(=O)(CC1CCc2ccccc21)N1C(CNC(=O)C#CC2CCOCC2)CC1 3700,c1(C(=O)NCCn2cc(C(=O)NC3CC3C(F)F)cn2)cc2cc(Cl)cnc2o1 3701,CC1CCCN(C(C2(CC3CCC3)CC2)=O)C1CCNC(=O)CCc1cccs1 3702,N(C1CN(C(C2(c3ccsc3)CC2)=O)Cc2ccccc21)C(c1c(C)ocn1)=O 3703,Cc1cc(F)cnc1C(c1nnnn1C1CCCCCC1)NC1CC(F)(F)C1 3704,C1(NC(CCC=C)=O)CC2C(NC(=O)C(C)(C)n3cnnn3)C2C1 3705,c1(N2CCC(NC(c3n(C(C)C)ncc3)=O)C(C)C2)nc2ccc(Br)cc2o1 3706,c1(C2(CN(CCNC(C3NC(=O)C4CC34)=O)CC3CC3)CCCC2)ncccc1F 3707,C1(C(=O)NCC(F)F)(CNC(c2c(CC)cns2)=O)CC(C)(C)C1 3708,Cn1ncc(C(=O)NCCOC(C)(C)CNC(=O)CC2C(C)(C)C2(C)C)c1Cl 3709,n1(NC(=O)NCC2(O)C(SCC)CC2)ccc(Br)cc1=O 3710,CC(C)(C(=O)NC1(C)CN(C(=O)CCOCC(F)F)C1)c1cccnc1 3711,N1(C(C2(C#C)CC(=O)C2)=O)CCCC(CC(=O)NCC(C)C(=O)OC)CC1 3712,C=CC(C)(O)CC(=O)NC(C)(CNC(=O)COCc1ccncc1)CO 3713,N1(C(C(CC)C2CCC(=O)N2)=O)CCC(O)C(N(C)C(C2CNC(=O)N2)=O)C1 3714,C1(C(=O)NC23CC(OC)(C2)C3)CCN(C(=O)C(C(=O)OC(C)(C)C)C2CCC2)C1 3715,C(=O)(CCS(=O)(=O)N(C)C)N1CCCC(CN(C(=O)C(Cl)=CCl)C)C1 3716,O(NC(=O)C(C(C)NC(c1cn2c(n1)CCC2)=O)C(C)C)C(C(=O)OC)(C)C 3717,CC(C)(C)C(C(=O)NC1CCN(C(C2CCCCNC2=O)=O)CC1)NC(N)=O 3718,N1(C(C=CC(C)NC(C=Cc2cc(C)no2)=O)=O)CC(CN(C)C)CC(C)(C)C1 3719,C(CCC(C)C)(C(=O)N1CCC(O)(CN(C(=O)CC2CCC2)C)CC1)NC(C)=O 3720,N1(C(C2CCN(C)C2)=O)CC2(CCC(CNC(=O)C(C)(C)C(C)(F)F)O2)C1 3721,c1(CN2CCC(C(=O)Nc3cc(SC)n[nH]3)C2)ccc(O)nn1 3722,c1(C(N(CC(F)(F)F)C)=O)cc(O)c2c(-c3ccc(OC(F)F)cc3)nn(C)c2c1 3723,c1(C(N2CC(COC)(CNC(=O)CNS(C)(=O)=O)C2)=O)cc(F)cc(F)c1O 3724,N#Cc1cc(F)ccc1-c1cn(C2CN(C(=O)CCCN3CCOCC3=O)C2)nn1 3725,N1(C(C23CCC(OC)C2C3)=O)CC2CCCC(C1)N2C(C1CC1Cl)=O 3726,c1(OC)ccc(C)cc1NC(C1CCN(C(=O)C2=COCC2)C1(C)C)=O 3727,C=CC1(C(N2CCN(C(c3cc(C)ns3)=O)C(CCC)C2)=O)CCOCC1 3728,CC(CC(=O)N1CCCCC1C(N)=O)C(C)(C)NC(=O)Cn1cnnc1O 3729,C(=O)(CC(C)(CN(C)C)C(F)(F)F)N1CCC2CN(C(CCC(=O)NC)=O)C2C1 3730,N1(CC(=O)N(C(C)CCO)C)CCN(C(=O)C(c2cnn(C)c2)O)CC1 3731,c1(CCC(=O)NC2(CNC(c3cc(C)nc(C)n3)=O)CC2)cc2ccccc2[nH]1 3732,c1(C(=O)NC(CC)CNC(=O)C(c2ccc(F)cc2)CC)ccc(OC)nc1C 3733,c1(C(=O)NC(C(=O)N(CCC(=O)OCC)C)C2CCCC2)cc(CC)c[nH]1 3734,C=CCCN=C(NCc1cc(Cl)cc(Cl)c1)NC1CCOC(c2nccn2C)C1 3735,C1(NC(C2(Cl)CCCNC2)=O)CCOC2(CCC2)C1 3736,C=CC1CCN(C(C2(n3cc(C(c4n[nH]cc4C)NCC)nn3)CCNC2)=O)C1 3737,c1(OC)ccc(CNC(=O)CC(C)N(C(=O)CC2CCCC(O)C2)C)nc1 3738,C(=O)(CC(C(F)(F)F)c1ccon1)NCCN(C)C(C1CCC(=O)NC1)=O 3739,Cc1nsc(N2CCN(C(=O)C(CCSC)NS(=O)(=O)c3cccs3)CC2)c1C#N 3740,N1(C(CCC(=C)C)=O)CCC(F)(CNC(C2CCC(=O)N2C2CC2)=O)CC1 3741,C1(CCNC(C(C)NC(C=CCOC)=O)=O)CCN(C)C1 3742,CC1CN(C)CC(C(=O)NC(C)C(N2CC(O)(CC(N)=O)C2)=O)O1 3743,CCC(CC)C(=O)NC1CCC(NC(=O)CNC(=O)CCC2CC2C)C1 3744,C123COC(C1)(C2)Nc1ccc(cn1)N(C(C)=O)C3=O.c1(COC)ncoc1C 3745,c1(CC)ccc(C)c(C(N2CC3(C2)CN(C(=O)C(c2ccc(Cl)s2)C)C3)=O)c1 3746,N1(C(c2c(OC)n(C)nc2C)=O)C2CCC1CN(C(C1CCCN(C(C)C)C1)=O)C2 3747,c1(C(=O)NCC2N(C(C3(C)C=CCC3)=O)CCC2)ccc2ocnc2n1 3748,C12(NC(C(CCSC)OC)=O)CC1CN(C(=O)Cc1ccccc1Cl)C2 3749,c1(C(N(C2CC3CC2CN3)Cc2cn(C)nc2)=O)cc(Br)cnc1O 3750,c1(CC(N2CC(O)(CN(C)Cc3ccon3)C2)=O)cnccc1C(=O)O 3751,c1(C(=O)NCCCC2(NC(C3C(C)CCS3)=O)CC2)ccc(OC(F)(F)F)cc1 3752,c1(OC)cccc(OC)c1C(=O)NCCC1CCCN(C(=O)C(C(C)C)OC)C1 3753,c1(OC)ccc2nc(N3CCC4(CCC(NC(=O)COC5CC5)O4)CC3)sc2c1 3754,CN1C2CCC1CC(=CC(=O)NCC1CCN(C(c3ccnnc3O)=O)CC1)C2 3755,c1(C(=O)NCC2CCC(C(N(CC=C)Cc3ccco3)=O)O2)c(C)noc1C 3756,c1(-n2cc(CCN(C(=O)C(C)O)CCOC)nn2)ccc(C(F)(F)F)cc1 3757,c1(C(N2CC(NC(=O)C3=COCC3)C3C2C3)=O)cc2n(n1)CCNS2(=O)=O 3758,CCC(C)(C)CC(=O)NC1(CO)CCN(C(c2csc3cncn23)=O)C1 3759,C1(CC(=O)NCCC2CCCO2)COCCN1C(c1nocc1Cl)=O 3760,c1(C(N(C2CCN(C(=O)CCC3CCCC3)C2)CC)=O)ccc2nc(O)[nH]c2c1 3761,C1(C(N2CCC(OC)C2)=O)C2C(CN1Cc1cccc3nscc13)C2(C)C 3762,c1(C(=O)NCC2(CNC(CCC(=O)OCC)=O)CC2)ccc(C)cc1OC 3763,C(=O)(C1CCc2c[nH]nc21)NCC1(C)CCN(C(C(CCCC)O)=O)CC1 3764,C1(NC(C2(C)CN(C(C(C=CC)O)=O)C2)=O)CNC(=O)OC1 3765,c1(C(N2CC(C)CCC2C)C(=O)NC(CC)C)ccc(F)c(C)c1F 3766,N1(C(C2CC(C)N(C)C2)=O)C2CCC(C(=O)NCC3CCC3(F)F)C1CC2 3767,C1(F)(NCc2cnc(NC(CN(C)C)=O)s2)CCN(C(=O)OC(C)(C)C)C1 3768,c1(SC)ccc(OCC(=O)NC(C)CN(C)C(c2ccc(F)s2)=O)cc1 3769,c1(C(N(CCNC(=O)C(C)S(N)(=O)=O)CC)=O)c(OC)ccc(F)c1N 3770,C(C(CC(C)C)C(=O)NC1CN(C(=O)Cc2coc3ccccc23)CC1O)OC 3771,c1(OCC)cc(OC)cc(S(=O)(=O)NCC(c2ccncc2)OC)c1 3772,C#CCC1CC(=O)N1.C(=O)(CC(=O)OCCC(=C)C)OC(C)(C)C 3773,Cc1nn(C)c2nc(C(=O)NCC3(CNC(=O)Cn4cnnc4O)CC3)ccc12 3774,C1(C(=O)NCCC(CC)(F)F)CC2(CCN(C(=O)C(O)CC(C)(C)C)C2)C1 3775,CCCC(CC1CCCCC1)C(=O)NC1CCCC1NC(c1coc(C)c1)=O 3776,C1(NC(c2cn(CCNC(C(C(C)(F)F)F)=O)nn2)=O)CCn2nnnc2C1 3777,c1(C(N(CC(C)NC(=O)CC(C)C(=O)OC)CC)=O)ccc2ccnc(O)c2n1 3778,Cc1cc(C(=O)NC2CCC2NC(=O)C(C)N(C)C)ccc1O 3779,CC1(C)COC(C(=O)NC2(CO)CCN(C(=O)COc3ccc(F)nc3)C2)CO1 3780,C1(NC(CC(c2cccs2)NC(C)=O)=O)(CN(C)C)CCN(C(=O)CO)C1 3781,c1(CC)cc(C(=O)NCCCCNC(c2ccnnc2)=O)c2c(c1)CCO2 3782,c1(OC)cc(NC2CCN(C(C3CC4CCCC(C3)C4)=O)CC2)ccc1[N+](=O)[O-] 3783,C1(C(N(CCOC)C2CC2)=O)CN(C(=O)C(C)C(F)F)CCO1 3784,Cc1ccc(C(=O)NCC2CCN2C(C2(O)CCCCCC2)=O)cc1C#N 3785,C(c1cccc(F)c1)=C(C(=O)N(CC(C)O)CCNC(=O)CC1(O)CCCC1)F 3786,c1(NC(=O)OCC)ccc(C(=O)NCC(C)(CO)NC(=O)CCC(C)C)cc1 3787,C(C)(CC(C)(C)O)NC(C=C(C)CNC(C1CN(C(C)C)C1)=O)=O 3788,CC1CC2(CCN(C(C3(c4cc[nH]n4)CC3)=O)CC2)CN1C(=O)CCC(N)=O 3789,C1(C(=O)NC(C)Cc2ccccn2)C2CC1N(C(=O)Cc1ccns1)C2 3790,C(CCCCc1ccccc1)(c1n(CCC)nnn1)NC(C)Cn1cncn1 3791,N1(C(c2ccc3nonc3c2)=O)CC2CCCC(C1)N(C(C1CC(O)C1)=O)C2 3792,c1(C(N(C)CCNC(C2(CO)CCOCC2)=O)=O)sc2cccnc2c1Cl 3793,N1(S(C)(=O)=O)C2CCC1CC(CN1CC3(COCCO3)C1)C2 3794,c1(C(N2CC3(N(C(CC=CCC)=O)CC3)C2)=O)ccc2ncn(C)c(=O)c2c1 3795,c1(CC(=O)OCC(=O)NCC(C(=O)OCC)C2CCOC2)ccc(OC)cc1Br 3796,N1(C(c2ccn(C(C)(C)C)c2)C(=O)NC2(C)CC2)CCC2C(C(N)=O)C2C1 3797,C1(NC(CCCOC(C)=O)=O)C2CC3C1C3C2C(=O)NC1(C)CCCC1C 3798,C1(NC(C)=O)CCN(C)C(c2ccccc2Br)C1.c12cc(Br)ccc1OC2 3799,C1(C(=O)NCCCCN=[N+]=[N-])CN(C(=O)CCOCC2CCC2)CC12CC2 3800,C=CCC(C(=O)NCC1CCC(C(=O)Nc2cccc(OCF)c2)O1)OC 3801,CC(C)C(O)C(F)(F)C(=O)NC(C1CC(NC(c2ccncc2)=O)C1)C 3802,n1(CC)c(C(C)NC(=O)N(C2CC3C=CN3CC2)C(C)C)nc2ccccc12 3803,C(N=c1[nH]c(N(C)Cc2ccc(Br)nc2)nc2c1CSC2)C1(OC)CCOCC1 3804,N1(C(C2N(C(C)=O)CCC2)=O)CCCCC1CCCNC(=O)CC1(CO)CC1 3805,CC1CN(CC(O)CNC(=O)C(=O)NC2CCCCNCC2)CC(C)O1 3806,C1(CCC(C)(C)NC(C2CCCC2(C)C)=O)CCCCN1C(=O)CSS(C)(=O)=O 3807,C(=O)(C(C)CC(=O)N1CC2CC2(NC(=O)CCCc2ccc(Cl)c(Cl)c2)C1)OC 3808,c1(C(=O)NCCCN2CCN(C(C3C(OC)CC3)=O)CC2)cccc(=S)n1O 3809,C1(CNC(C2C3CCCC23)=O)CCCN(C(=O)CCc2cnc(C3CCC3)s2)C1 3810,N1(C(C(C(C)C)OCC(C)C)=O)CCC2(CCN(C(c3ncc[nH]c3=O)=O)C2)C1 3811,c1(C(=O)NCC2CCN(C(C(F)OC)=O)C2)cc(C)cc(N)c1 3812,CC(C)(C)C(CC(F)(F)F)NS(=O)(=O)Cc1ccc(F)cc1Br 3813,Cc1ccc(CCC(=O)NC(C)CCNC(C2C(C)C2C)=O)c(C)c1 3814,C(C)(C(=O)N(C(C)C=CC(=O)NCCCO)C)SCC 3815,c1(C(=O)NCC(C)CNC(c2n[nH]c3c2CCC3)=O)cc(O)nc(Br)c1 3816,C1(C(N(CC(C)NC(=O)Cc2cc[nH]c2)C)=O)CC(=O)N(c2ccccc2F)C1 3817,CCC1=NOC(CC(=O)NCCC(C)N(C(=O)CSc2nccn2C)C)C1 3818,c1(C(N(C)CC2CCN(C(C=C(COC)C)=O)C2)=O)cnc(C)n1C 3819,c1(C(=O)NCC2CCC(NC(C3CC(C)N(C)C3)=O)C2)cc(Cl)ccc1[N+](=O)[O-] 3820,c1(C(=O)NC(CNC(C2N(C)CCC2)=O)(C)C)ccc2c(=N)[nH]cnc2c1 3821,CC(=O)CCCC(=O)NCC12CC(C1)C(NC(=O)CCOCC(F)F)CO2 3822,n1(CC)cc(C(N2CCOC(CCCNC(=O)C=C(C)C(C)(C)C)C2)=O)c(C)n1 3823,c1(NC(=O)Nc2c(SCC)cc(Br)cc2)ccc([N+](=O)[O-])cc1Cl 3824,c1(SC(C)C(=O)NCCC2CCN(C(=O)C=CCn3cncn3)C2)ccccn1 3825,c1(C(C)NC2(c3cn(-c4ccsc4C(=O)O)nn3)CC2)cc(C2CCC2)nn1C 3826,CCC(F)(F)C(C)(C)C(=O)NC(C)CN(C)C(c1cc[nH]c(=NC)c1N)=O 3827,c1(CC(=O)N(CC(=O)N(CCCO)CCO)CC#C)cncnc1 3828,c1(OC)ccc(COC2CC2C(=O)OC2(C)CCC2)c([N+](=O)[O-])c1 3829,C1(C(=O)NC(CC(=O)NCC(CCC)C)COC)CC2CC1CC2=O 3830,C(=O)(C1=CCCN(C(c2ccc(O)cc2Br)=O)C1)Nc1ccc(C#N)nc1 3831,CC1CN(C(=O)CSC(C)(C)C)CCC1CNC(=O)C(C)Oc1cccnc1 3832,c1(OC)cccc(C(N2CCN(C(C)CNC(=O)C(C)CS(C)=O)CC2)=O)c1C 3833,C#Cc1ccc(F)c(C(N2CCCC(CNC(C3CCC(=O)C3)=O)C2)=O)c1 3834,N1(C(CCC(=O)N(C)C)=O)CC2CCC1CN2C(C1CC2CC2CO1)=O 3835,CN1CC=CCC1CCC(N1CCC(CC(=O)NC(c2ccon2)(C)C)C1)=O 3836,N1(C(CCC=C)=O)CCCC(C2CCCN(C(=O)CCc3cncc(F)c3)C2)C1 3837,N1(C(C(C)N(C(C)=O)C)=O)CC(O)(C(C)NC(=O)Cc2cnsc2)C1 3838,CC1CN(C(=O)CC2C=CCC2)C1C(=O)NCC(C)(C)CC1CC1 3839,C#Cc1ccc(C(=O)NC2CCN(C(c3nscc3Br)=O)CC2O)cn1 3840,c1(C(N2CCC(O)(C(F)F)CC2)C(=O)NCCOCC)ccc2ccoc2c1 3841,c1(CCC(=O)NC2CCC3CC2CN3C(=O)CCF)cnc2n1CCCCC2 3842,N1(C(C(=O)NCCCOC)c2ccsn2)CCOC(c2cccs2)CC1.S(C)(=O)(=O)N 3843,c1(C(C)(C)C)cc(C(N2CCC(C)(NC(=O)Cc3ccoc3)C2)=O)ccc1O 3844,c1(OC)c(C(=O)NCCCNC(=O)COC(F)F)ncnc1C 3845,C(=O)(C(C)COC)NC(C(=O)N(CCC)CC1CC1)c1cccs1 3846,c1(OC)ccc(F)cc1CC1CCCCC1C(N1CCCC(Cn2cccn2)C1)=O 3847,C1(N(C(=O)C(O)CC)CCC)CCN(C(c2csc(C)c2Br)=O)CC1 3848,C12(CNC(C34CC(C)C3C4)=O)CC1CN(C(C1(CO)CC(C)(C)C1)=O)C2 3849,c1(C(N2CCC(F)(CNC(CCOCC#C)=O)C2)=O)cc2ccncc2s1 3850,N1(CCC)CCCC(CNC(=O)N(C)Cc2n[nH]cc2Br)C1 3851,N1(C(C(=O)NCC)=O)CCC2(CCCN2C(=O)C(O)CC(C)(C)C)C1 3852,n1(CCC(N2CC(CCNC(C3C(C)(C(C)C)C3)=O)C2)=O)ccc2cccnc12 3853,CC(C)CC(F)C(=O)NC1(C2CN(C(=O)Cc3cc(-c4ccco4)on3)C2)CC1 3854,C1(NC(=O)CCc2cccnc2)CC2CC(NC(c3ccc(Cl)[nH]3)=O)C2C1 3855,C=CCCC(C)NC(C1CCCC1CNC(C1CN(C)C1)=O)=O 3856,C1(CNC(C(COC)O)=O)C2CCCC1N(C(c1ccc(O)c(Cl)n1)=O)C2 3857,CC1(C)OCC2CC12C(N1CCN(CC(C)(C)NC(=O)CC2=CCCC2)CC1)=O 3858,Cc1nc(CNC(C2CCOC2C(C)C)=O)sc1CNC(=O)COCC1CC1 3859,c1(C(C(=O)NCC2CN(C(c3c(C)cco3)=O)C2)C)ccc(Br)c(C)c1 3860,C(=O)(CS(=O)C(F)(F)F)NC(CNC(c1c(CC)ocn1)=O)C1CCC1 3861,CC#CCC(C(=O)NC(c1nc(C)cs1)C)NC(=O)COc1cnn(C)c1 3862,CCCCCC(O)C(=O)N1CCC2CC12C(=O)NCc1ncnn1CCC 3863,N1(C(C(C=CC)O)=O)CC(CNC(C2C(Cc3ccccc3)CSC2)=O)CC1(C)C 3864,C(=O)(C(C(=O)NC(C)(C)C(C)NC(c1occc1CN(C)C)=O)OC)OCC 3865,c1(C(=O)NCCC2CCC(NC(COCCOC)=O)C2)cc([N+](=O)[O-])ccc1N 3866,C1(COCC(=O)NC2CCCOC2)CCCNC12CC2 3867,C1(CC=C)(NC(C2CCS(=O)(=O)C2)=O)CCN(C(C2CCCNS2(=O)=O)=O)CC1 3868,Cc1cc(C)c(C(=O)NCc2ccccc2C)c(Cl)n1.N12CCC(C1)NC2=O 3869,CC1(C)OC(=O)NC1CN(CCC1CCCCC1)C1CC1 3870,c1(C(C(=O)OC)NC(=O)C(F)CC(C)C)cccc(Br)c1OC 3871,Cc1onc(CO)c1C(=O)NCCCN(C(=O)C=C(Cl)Cl)CCO 3872,C(=O)(C(C)C(O)C(C)C)NC1(C(=O)NCC(CCOC)(C)O)CCSC1 3873,CC(C)C(C(=O)NC1CC(C(F)C(=O)NC2(CO)CCOC2)C1)c1cnn(C)c1 3874,C1(C(C)C(=O)NCC(=O)N(CCCO)C2CC2)CCC(=O)N1 3875,N1(C(CC2CN(C(c3c(CC)ccs3)=O)C2)=O)CCCCC1C1(COC)CC1 3876,CC(C)C(CCS(C)(=O)=O)NCC(=C1CCNCC1)F 3877,c1(OCC(=O)NCCCNC(CC(=C=C)C)=O)ccc(C)cc1C(C)(C)C 3878,C1(C(N2C(C)CC2NC(c2cc(O)n(C)n2)=O)=O)CCc2ccccc2C1 3879,C12(CNC(c3ccc(C(C)C)o3)=O)CC(CN1C(C1CCCCO1)=O)C2 3880,C1(CNC(COCCC)=O)CC2(CC2)CN1C(c1cn(C2CCOC2)cn1)=O 3881,Cc1ccccc1OCC1(C(=O)O)CC1(C)C(F)F.c1(N)nc(C)cs1 3882,c1(C(N(C)CC2CCCN(C(c3scc(C)c3Cl)=O)C2)=O)cc(O)nc(Cl)c1 3883,C=CC(C)(CC)C(=O)N(CCCNC(c1ccc(C(=O)OC)nc1)=O)CCO 3884,c1(NC(C2CC(F)CN2C(c2ccc(C3CC3)cc2)=O)=O)ccnc(C2CC2)c1 3885,C12(CNC(c3cc(C)nnc3)=O)CCC1CCN2C(=O)CSC(F)(F)F 3886,C(=O)(CCCCN=[N+]=[N-])N1C(C(=O)NC(CC=C)C(=O)OC)CC1C 3887,C1(CCC)(C(=O)NCC(c2cccc(Cl)c2)NC(c2ccco2)=O)CCNC1=O 3888,Nc1cccnc1C(=O)NCC1CCCCC1C(=O)NCc1ncc(CO)[nH]1 3889,C(=O)(CC(C)C(F)F)NC(C(=O)N(CC(CC)(O)CC)C)COC(C)C 3890,C=CCC(CNC(C1(CO)CCCC1)=O)NC(C1(c2ccno2)CCC1)=O 3891,C1(NC(Cc2nn(C)nc2Br)=O)CN(C(C2CCCN2C=O)=O)CCC1CO 3892,C(CC(C(=O)N(C(C)CCNC(c1cocn1)=O)C)OC)OC 3893,c1(C(=O)NCC2(C#N)CCC2)c(NCC2CCC(C(N)=O)O2)sc2c1CCCC2 3894,C=CCC(C)(CNC(=O)CC1(C)CCN(C(=O)COCCC)C1)CO 3895,c1(COC)cccc(C(=O)N(C)CCN(C(=O)CCc2ccn(C)n2)C)c1 3896,C#CC1CCCN(C(=O)C(=O)NCC2COC3(CCCC3)C2)CC1 3897,N1(C(C(COCC)C)=O)CCSCC1C(=O)Nc1ccc(Cl)nc1 3898,C1(NC(C2(OC)CC2)=O)CC(O)CN(C(c2cnc(C3CCC3)s2)=O)C1 3899,C1(COCC(=O)NCC2CC(NC(c3cc(Cl)no3)=O)C2)CCCCO1 3900,Cc1nsc(NC(C2CCN(C(=O)CCC3(O)CCC3)CC2)C)c1C#N 3901,N1(C(C2CN(C)CC2C(F)(F)F)=O)CCCC(NC(C2(CO)CCC2)=O)CC1 3902,Cc1nccn1CC(=O)NC1(C(=O)NCC(c2ccco2)O)CCSC1 3903,C1(N(C(C=C(CC)C)=O)C)CCCCN(C(c2cn(C)c(O)n2)=O)C1 3904,Cc1c(F)cc(CN2CCN(C(=O)Cc3ccc(F)cn3)C(C)C2)cc1F 3905,N1(C(C2C(NC(c3[nH]cc(C(C)(C)C)c3)=O)CCC2)=O)CCOC2CC12 3906,C1(C(C)O)COCCN1C(c1sccc1CNC(C1CCCNC1=O)=O)=O 3907,c1(OC)cc(-c2nc(CCCOC(C)C)nn2Cc2cccc(C)c2)n(C)n1 3908,c1(C(N(CCN(C(C(C)OCC)=O)C)C)=O)cc(Cl)cnn1 3909,CC1=CCC(C(=O)NCCC(C)NC(=O)CSc2cccc(F)c2)CC1 3910,C1(C(C)C)CCCN(C(=O)N(C(C2CCC2)=O)Cc2nc(C(=O)O)n[nH]2)CC1 3911,c1(N2C3CCC(C(NC(C)=O)C2)C(F)(F)C3)ncnc2ccc(F)cc12 3912,N1(C(CC=C)=O)CCCC(CC)C1C(N1CCC(CCOC)CC1)=O 3913,C(C(C)(C(=O)N(C1CCCC1)C)NC(=O)CC1CC(=O)NC1=O)SC 3914,S(=O)(=O)(c1ccccc1NC(=O)N(C)CC1(O)CCC(C)(C)C1)N(CC)CC 3915,C(=O)(CCCCCCCCCO)NC(CNC(C1C(=C)CC1)=O)CO 3916,C1(C(=O)NCC(C)CNC(=O)COCC2CC2)CCS(=O)(=O)C1(C)C 3917,C#CC1CN(C(=O)C(CCOC)NC(c2cnns2)=O)CCO1 3918,N1(C(C2(CC#C)CCOC2)=O)CCC2(CC(NC(=O)C(C)(C)CF)C2)C1 3919,c1(OC)cc(F)c(NC(=O)C(=O)NCC2CNCC2C)c(F)c1 3920,c1(CC)ccccc1C(=O)Nc1ccco1.C12CCCC1n1cc(nn1)CN2C 3921,C1(C(N2C(CNC(CC(CC)OC)=O)CC2)=O)CNc2ccnn2C1 3922,C#CCC(CC#C)C(=O)NCC1CCCC(NC(=O)Cc2cc(C3CC3)on2)C1 3923,C1(C(=O)NC(CNC(C(C)c2ccsc2)=O)C2CC2)Cc2nccn2C1 3924,C1(NC(CC2(NC(C)=O)CC2)=O)CCCN(C(=O)C(F)(F)C2CC2)CC1 3925,Cc1nnc2ccc(C(N3CCCC3CNC(c3occc3F)=O)=O)cn12 3926,Cc1c(F)ccc(C(=O)NCC2CC2CNC(C2CCS2(=O)=O)=O)c1Cl 3927,c1(OC(CNCC(C)CO)(C)C)cccc([N+](=O)[O-])c1 3928,CCC(O)C(C)C(=O)N1CC(CNC(C2CCS(=O)CC2)=O)C(C)(C)C1 3929,C1(CC(C)C)C(=O)NCCN1C(=O)NC(c1ccc(F)cc1Br)C 3930,C1(CNC(C#CC(C)C)=O)CC2(CCOCC2)CN1C(=O)CC1CC(=O)NC1=O 3931,N1(C(C2C(CC)CCC2)=O)CCN(C(c2ccc(NC(C)C)cc2)=O)CCC1C 3932,c1(CCC(=O)NC2(CNC(=O)C(O)C3CC3)CC(OC)C2)cccnc1Cl 3933,O=C(CCCNC(C1CC=CCC1)=O)NCC1C=CCN1C(=O)CC1CSC1 3934,C1(C(C)NCC(c2ccccn2)CN)CCCN(Cc2ccccc2)C1=O 3935,C(C)(CC(C)(C)CO)NC(C(C)(C)NC(C=C(CCC)CCC)=O)=O 3936,CC(C)(CC#N)C(=O)N1CCCC(NC(c2ccc(F)c(CO)c2)=O)C1 3937,c1(C(=O)NCCCN2CCC(NC(C3(C#C)CCC3)=O)C2)cc(O)ccc1C 3938,CCC(CC(=O)NCC12CC(CCO1)C2)NC(=O)C(CCSC)OC 3939,C1(NC(c2c(C)nc(CO)s2)=O)CN(C(=O)C2=CCCOC2)CCC1C(F)(F)F 3940,Cn1ncc2c1CCC(C(N1CCN(C(=O)Cc3cc(C4CC4)on3)CC1)=O)C2 3941,N1(C(C(c2ccncc2)C)=O)CCC(O)(CCNC(=O)Cc2n[nH]c(=N)s2)CC1 3942,CC(N=c1[nH]c2c(c(=NCCC3CCOC3)[nH]1)CCCC2)C1CCCC1 3943,O=C(CN=c1cc(F)nc(-c2ccccc2)[nH]1)C1CC2(C1)CC(F)(F)C2 3944,C1(NC(C=C(C)C(C)(C)C)=O)CCCCCN(C(=O)COC2CCN(C)CC2)C1 3945,C=Cc1cc(C(=O)N(CC(N2CCC(C(=O)NC)C2)=O)CC)cc(F)c1 3946,c1(C(N2CC(CCC)N(C(c3ns[nH]c3=O)=O)CC2)=O)c(F)ccc(F)c1F 3947,c1(OC)ccc(F)c(CC(=O)N(C2CN(C(c3ncccn3)=O)CC2(C)C)C)c1 3948,N1(C(CC(C=C)(C)O)=O)CCCN(C(=O)CC23CCC(CC2)C3(C)C)C(CO)C1 3949,C1(NCC2(CC#N)CCC2)CCNC(c2ccccc2)C1 3950,C=CCCC(O)CNC(=O)CC(O)CNC(c1csc(C)c1C)=O 3951,C1(NC(C(Cc2ccco2)NC(COCCCCC)=O)=O)CCCC2(CCC2)C1 3952,Cc1sc(C(=O)NCCC2CCCN2C(C2CC23CCC3)=O)cc1CS(C)(=O)=O 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3989,N1(C(c2c(O)ccc(C)c2)=O)C2CCC(C(N3CCC(O)(CO)C3)=O)C1CC2 3990,N(C1CCCc2sccc21)C(N1CC(CC2CCOC2)C1)=O 3991,C(=O)(C(CC(F)F)NC(=O)OC(C)(C)C)N1CC(N(C)C(C2CC=CCC2)=O)C1 3992,c1(C(=O)NCCCCCCNC(c2sc(C)c(O)n2)=O)cc(Cl)ccc1F 3993,N1(CC)Cc2cc(CNC(c3cc4cccc(F)c4[nH]3)C)ccc2C1=O 3994,C1(CNC(C(C(CC)C)O)=O)CC2(CCN(C(=O)Cc3cnc[nH]3)CC2)C1 3995,C(=O)(C(CCSC)NC(=O)C(Cl)Cl)NC1(CC=C)CC1 3996,N1(C(CN(C(=O)OC(C)(C)C)CC)=O)CCC(CC(C)NC(=O)C(F)CC)CC1 3997,CCCC(C(=O)N1CC(NC(=O)COCC(F)(F)F)C1)OC.C12CCN(C1)C2 3998,C1(C)(C(N2CC=CC(NC(c3c(OC)nn(C)c3)=O)C2)=O)CC(O)CN1C 3999,CCC(CC1CCCC1)C(=O)NC1CN(C(c2sc(CO)nc2C)=O)C1 4000,c1(C(=O)NC2C(NC(c3cn(C)nc3)=O)CCCC2)cnc2[nH]cnc2c1 4001,C1(NC(c2cncc(O)c2Cl)=O)CCCCN(C(C2CCC(F)(F)CO2)=O)C1 4002,C1(NC(c2ccco2)=O)CN(C(C2CNCC3(CCC3)O2)=O)C2(CCC2)C1 4003,CCCC(C(=O)N(C1CCN(C(c2ccc3nn[nH]c3n2)=O)C1)CC)S(N)(=O)=O 4004,CC(F)(F)C(C)(C)C(=O)N1CC(CCCCNC(c2ccc(C(N)=O)o2)=O)C1 4005,c1(C(=O)NC2C(C)CN(C(=O)C(C)Sc3ccccn3)C2)nnn2c1CCCC2 4006,C1(CNC(C(CC)O)=O)CC12CCN(C(c1n[nH]c3c1COC3)=O)CC2 4007,O=C1CCC(C(=O)NCCC2CCCCN2C(c2ccsc2C(F)F)=O)CN1 4008,c1(C(N(CCNC(C2C(CC)CCO2)=O)CC)=O)[nH]c2ccc(F)cc2c1C 4009,CCCC(C(=O)N(C)CCN(C)C(c1cc(F)ccc1Br)=O)C(C)C 4010,c1(C(N2C(CNC(c3ccns3)=O)CC(OC)C2)=O)cc(Cl)c(F)cc1O 4011,Cc1ccc(OCCC(N2CC(NC(=O)CCC(C)C#N)C3(CC3)C2)=O)cc1C 4012,CCCC(C(=O)N1CC(NC(N)=O)C1)c1ccc(Cl)cc1 4013,c1(OC)cncc(Br)c1C(=O)NC1CC1CNC(=O)CC1CCCCC1 4014,CC(C)(C)CC(O)CC(=O)NC1CCCC1C(=O)NC(CCO)C(F)(F)F 4015,CCCC(C(=O)NCC12CC1CN(C(c1cnccc1Cl)=O)C2)OC 4016,c1(C(C)OC)nc(C(=O)NC(CNC(c2cn(CCF)nn2)=O)CO)co1 4017,c1(C(N(C2CCCN(C(C(CC)O)=O)C2)C)=O)cc(O)cc(N)c1Cl 4018,N1(C(C2C(OCC)CC2)=O)CCN(C(=O)C=CCNC(C)=O)CC1C 4019,c1(CC(=O)NC2C(NC(c3cc(C)on3)=O)CCC2)c(C)[nH]c2ccnn2c1=O 4020,CCCCC(CC)C(=O)NC(CNC(c1ccc(CCC#N)cc1)=O)CC(C)C 4021,C1(C(N2C(C3(NC(C4(CCCC)CC4)=O)CC3)CCC2)=O)CC(O)CN1C(C)=O 4022,Cc1nnc(O)c(C(=O)NCCC2CSCCN2c2ncc(Br)cn2)c1C 4023,c1(C(=O)NCC2(N3CCOCC3)CCCOC2)nc2ccc(F)cc2s1 4024,c1(C(N2CCCC3(NC(C(C)C)=O)C(C2)C3)=O)n[nH]c2ccc(Br)cc12 4025,c1(C(C)NC(C2CCCN(C(=O)COC3CCCCC3)C2)=O)cc(Br)ncc1F 4026,c1(C(N(C2C3CN(C(C(C4CCOCC4)OC)=O)CC32)C)=O)ccc(Cl)c(F)c1 4027,N1(C(c2ccc(F)c(Cl)c2)=O)CC2CCC1CN2C(C1SC2C=CC1CC2)=O 4028,N1(C(C2C(C(=O)OCC)C2)=O)CSCC1C(=O)NCC=Cc1ccco1 4029,C1(C(=O)NCCCC(C)NC(C(C)NS(C)(=O)=O)=O)CC2(C1)CC2F 4030,Cc1ccc2ccccc2c1CNC(c1sc(CC2CC2)nc1C)C1CC1 4031,c1(N2CCC(N(CC#C)C(c3cscc3C)=O)CC2)ncnc2cc(Br)sc12 4032,C1(NC(C(C)N(c2ccnn2CC(F)F)C)=O)CC(C)(NC(C2CCCC2)=O)C1 4033,C1(CC(N2CCCC(NC(C3CC3C3CCCC3)=O)C2)=O)CCCCC1(F)F 4034,C1(N(C(c2ccoc2C2CC2)=O)C2CC2)C=CCN(C(=O)COCC(F)(F)F)C1 4035,C(=O)(C(O)CC(N)=O)NC(C)CCC(=O)NCCc1cccc(O)c1 4036,CC1CCC2(CC1)CCN(c1nnc(-c3nc(Br)cs3)n1CC1CCCCO1)C2 4037,c1(C(=O)NCC2CCC(NC(C(CC)(C)CO)=O)C2)n[nH]c2cccc(OC)c12 4038,C1(C(=O)NC(CNC(C(CC)=CC)=O)(C)C2CC2)CCc2cn(C)nc2C1 4039,C1(NC(Cn2ccc(C)n2)=O)CCN(C(C2CC(n3cnnc3)C2)=O)CC1F 4040,C(=O)(CCC(=O)N(C)C)N(C(C)C)C1CC1.C12COC(C1)CNC2=O 4041,C1(NC(C2CN(S(CC)(=O)=O)C2)=O)(CO)CN(C(C2(C#N)CC2C(=O)NC)=O)C1 4042,c1(C(=O)NCC2CC(CNC(CSCCCC)=O)OC2)onc2c1CCCC2 4043,C(CCC(C(=O)Nc1ccccc1)N(C1CCN(C)CC1C)C)=C(C)C 4044,CCC(C)CC(C(=O)NCc1cc(C#N)n(C)c1C)NC(C)=O 4045,C(=O)(CC(F)(F)C(F)F)N1CCCN(C(C(c2ccc(OC)cc2)C)=O)CC1 4046,c1(CC)ccc(CC(N2CCOCC2c2cn(-c3ccc(Br)cc3)nn2)=O)cc1 4047,c1(OC)noc(C)c1C(N1CCC(C(C)NC(=O)CC2(C)CCCCC2)C1)=O 4048,N1(C(C(C2CN(C(C(C=CC)O)=O)C2)O)=O)CC2(C1)CC2(F)F 4049,C(=O)(C(CC(C)C)NC(c1cnc(Cl)n1C)=O)NCC1CC(CC)C1 4050,N1(C(C(CC=C)CC)=O)CCC(C2(NC(=O)COC3CC(F)(F)C3)CC2)CC1 4051,c1(C(=O)NC2(C)CN(C(C3CCOC(=O)N3)=O)C2)cc2c(nc1O)CCCCC2 4052,c1(C(=O)NCC2C=CCN2C(C2CCCC2(F)F)=O)ccc2c(n1)OCCO2 4053,C1(O)(CCNC(CSCCCC)=O)CCCN(C(=O)CCn2cccnc2=O)C1 4054,C1(NC(C(C)N(CCSc2ccccc2)C)=O)CN(C(=O)C(=O)N(C)C)CC1O 4055,c1(C(=O)NCCCCCN(C(c2cc(SC)c(C)o2)=O)C)nc[nH]c2ncnc1-2 4056,c1(OC)ccc(Cl)c(C(=O)NCC23CC2CN(C(=O)CC(C)(C)OC)C3)c1 4057,N1(CC#CCOC)CCC2(CCN(C(c3csnc3OC)=O)CC2)C1 4058,c1(C(N2CCCC(N(C(C3C=CCCC3)=O)CC3CC3)C2)=O)cnccc1Cl 4059,C1(CNC(c2n(CC)ccn2)=O)CCN(C(C2CSC(C)=N2)=O)C12CCC2 4060,N1(C(CC(N)=O)=O)CCN(C(=O)CSC2(CC#C)CCCOC2)C(CC(F)F)C1 4061,C(C(CC(F)(F)F)NC(=O)Cc1cc(F)cc(F)c1)NC(C(CC)NC(C)=O)=O 4062,C12CC(CCO1)NC(=O)CCN(C)C2=O.c1(CC)cnccc1C 4063,C(CCC(C)C)(C(=O)NCCc1nccnc1C)NC(c1c(CC)c[nH]n1)=O 4064,C(=O)(C(C)(O)C(F)(F)F)Nc1ccc(C)c(Cl)c1.C=C1CNCC1 4065,c1(-c2nc(OCC(N3CCC(CS(N)(=O)=O)C3)=O)sc2)nc2ccc(F)cc2s1 4066,Cc1ccc(C)c(CN2CCC(C)(C(=O)NC3CCN(S(C)(=O)=O)C3)C2)c1 4067,C1(C(N(C)CCN(C(=O)C(C2CCCO2)C2CC2)C)=O)CCCC2C1C2(F)F 4068,N1(CC(=O)NCC=C)CCCC(CO)(NC(C2CC2C)=O)C1 4069,C(=O)(C(C1=CCCSC1)N1CCOC(C(C)(C)C)C1)NCC=C 4070,C(N=c1ncc([N+](=O)[O-])c[nH]1)C1CCC(NC(c2nc(C(C)C)sc2)=O)C1 4071,N1(C(c2c(N)cc(F)cn2)=O)CC=C(CC(=O)NC2CC2O)CC1 4072,C1(C(=O)NC2CN(C(c3c(CCC)occ3)=O)C(CO)C2)CC2(CC(OC)C2)C1 4073,C(CCC(C)(C)CO)NC(C1CC(NC(CC2ON=C(C)C2)=O)C1)=O 4074,C1(NC(c2c(CC)cno2)=O)CS(=O)(=O)CC1NC(c1cnc(C(C)C)nc1)=O 4075,C(C(C)(CO)CO)N(C(=O)C(C1CC1)N(C(=O)CC(=O)N(C)C)C)C 4076,C1(C(N(C)CC2(N(C)C)CC2)=O)CN(C(=O)CCn2cnc(=N)[nH]2)CC1(F)F 4077,c1(NC2CC(C(=O)Nc3nc(C)c(C#N)nc3)C2)ncnc2sc(Br)cc12 4078,c1(CNC2CC(NC(CNC(CC(C)C)=O)=O)C2)cc(F)cc(Cl)c1 4079,N1(C(CCCSC)=O)CC2CCC(NC(c3ncoc3-c3ccon3)=O)CC2C1 4080,c1(C(=O)NCCNC(C2CCN(C)C(=O)C2)=O)cccc2ncccc12 4081,N1(C(N2CC(C)C(NC(=O)OC(C)(C)C)CC2)=O)CCOCC(F)(NCO)C1 4082,c1(C2C(C(=O)NC(CC)CN(C(=O)Cc3ccc(C)s3)C)C2)ccccc1C 4083,C1(F)(C(N2CCC(CN(C)C(C3(CF)CCOCC3)=O)CC2)=O)CCS(=O)(=O)C1 4084,C1(C(N(C(C)CNC(C2CCCC2)=O)C)=O)CCCSC1 4085,N1(C(C=CC)=O)CC2CC(NC(=O)C(C3CCC3)OC)CC1C2 4086,N1(C(C2CC(CNC(C(C(C)C)OC)=O)C2)=O)CC(CO)CC12CCC2 4087,c1(CSC)cc(C(=O)NC2CCC2CNC(c2cc(Cl)no2)=O)ccc1F 4088,Clc1cc(Br)ccc1-n1nnnc1CNc1ccccc1C1CCNCC1 4089,N1(C(CN2C(C)CCC2C)=O)CC2(CCC(CNC(=O)C(C)N3CCCC3)O2)C1 4090,C1(C(=O)NCCNC(C=C(C)C(C)C)=O)CCCOC1c1cn[nH]c1 4091,C12(NC(=O)Cc3ccoc3)CCCC1N(c1cc(Cl)nc(C(F)(F)F)n1)CC2 4092,O(N1CCC(N=c2cccc(S(=O)(=O)N3CC(C)OC(C)C3)[nH]2)CC1)CC 4093,c1(OC)ccc(Cl)c(C(=O)N(C2CCCN(C(=O)C(C)OC3CCCC3)C2)C)n1 4094,C1(NCC2CCCC(CNC(C(n3cc(CO)nn3)C)=O)C2)CCC(O)CN1C 4095,C12(CNC(=O)CO)CC(NC(=O)C(c3ccccc3)O)(CO1)C2 4096,C1(CCNC(c2c(CNC(C(COC)C)=O)ccs2)=O)OCCC1(C)C 4097,c1(C(N2CC3(CNC(C=C(C)Cl)=O)CC(F)(C2)C3)=O)cnc2c(C)cccn12 4098,Cc1cc(CNc2cc(F)cnn2)cc(C(F)F)c1 4099,C1(CCNC(C2N(C(CC)=O)CSC2)=O)COCCN1C(=O)COC1CC1 4100,N1(C(C2(C)CC(NC(C3CCN(CC)C3)=O)C2)=O)C2CSCC1C2 4101,Cc1cc2c(Br)n[nH]c2cc1NC1CCCC(O)(C(F)(F)F)C1 4102,c1(OC)ncc(NC(=O)CC(CNC(=O)C(N2CCNC2=O)C)OC)cn1 4103,Cc1cc(Br)cnc1C(=O)NC(CNC(=O)COC(F)(F)F)C(C)(C)C 4104,c1(C(=O)OC)nc(Cl)c(Cl)c(NC(=O)C(=O)N(C)CCOc2ccc(F)cc2)c1Cl 4105,CC1=C(C(=O)N2CC3CCCC3(NC(=O)Cn3cc([N+](=O)[O-])cn3)C2)CCCO1 4106,c1(C(N(CCN(C(=O)CC(=O)NC2CC2)CC)CC)=O)ncsc1C 4107,c1(NCC(=C)C2CCOCC2)ccc(S(=O)(=O)NC2COC3(CCCC3)C2)cn1 4108,Cc1nc(N2CCC3(NC(=O)C4=NNC(=O)CC4)CCCC23)c2ccsc2n1 4109,C1(C)(C(=O)NC(C2OCCN(C(CCCOC)=O)C2)C)CC(C(C)(C)C)=NO1 4110,C1(C(N(C2CCCC(NC(C(C)OCCC=C)=O)C2)C)=O)C2CC3C(C2=O)C13 4111,N1(C(c2nc(C(C)NC(CSCC#C)=O)oc2)=O)CCC2(CCCN2C)C1 4112,c1(CNC(CSCC)=O)ccccc1CNC(c1ccsc1CC)=O 4113,Cn1cnc(C(=O)NC2COCCN(C(=O)CNC(c3cscn3)=O)C2)cc1=O 4114,c1(C(=O)NCC2CCCC(NC(C(CC)(C)CO)=O)C2)ccc2cnoc2c1 4115,Cc1ncc(N)cc1C(=O)N(CC(C)NC(=O)C(C)NC(=O)Nc1ccco1)C 4116,Cc1cnc(CNC(=O)CCCC2CN(C(=O)OC(C)(C)C)C2)o1 4117,Cc1nc(SCc2ncc(CO)s2)c2ccccc2n1 4118,n1(CC)nccc1C=CC(=O)NC1CN(C(c2cn(C)nc2O)=O)CC1OC 4119,c1(C2CCN(C(C(c3ccc(Br)nc3)(C)C)=O)CC2)cccc(F)c1 4120,c1(C(=O)NC2C(C(=O)Nc3ccc(OC)cc3C)CCC2)cn2ncccc2n1 4121,C1(CC)CCOC1C(=O)N(CCC(=O)NCC1(O)CCCC1)C(C)C 4122,[N-]=[N+]=NC1CN(C(c2n[nH]c3c2COC3)=O)CC1NC(=O)C(C1CC(F)(F)C1)O 4123,Cc1ccc(C(N2C3CCC2C(NC(C2CC4CCC2C4)=O)C3)=O)cc1C 4124,C1(CCC(=O)N(CC=C)CCC)CCCN(C(=O)C(C)NC(C)=O)C1 4125,C(=O)(C1CC=Cc2ccccc21)NC1C2CN(C(C#CC3(C)COC3)=O)C(C2)CC1 4126,Cc1nc(CNC(=O)CCc2cccn2C)oc1C(=O)NC(C)Cn1cnnc1 4127,N1(C(C2CC(C(C)C)OCC2)=O)CCC(F)(CNC(C2C(C)C2C)=O)CC1 4128,c1(OC)cc(OC)cc(C(N2CC(NC(c3cc(C#N)oc3C)=O)C(C)C2)=O)c1 4129,C1(NC(C23CC(C)C2C3)C)CCN(CC2CCCO2)CC1 4130,Cc1ccc2c(C(=O)NCC3CC(NC(=O)C(=O)N(C)C)C3(C)C)csc2c1 4131,C(=O)(C#CC1(C)CCCO1)N1C(C(=O)NC2(CC=C)CCC2)(COC)C=CC1 4132,C=CCCC(C(=O)N1CCCC(O)(CC)C1)NC(=O)CN(C)CCOC 4133,C1(F)(C(=O)NCC(C2CCOC2)NC(c2ccns2)=O)C2CCCC12 4134,C1(C(C(=O)OCC)CC)CCN(c2nnnn2CC2CC2C2CC2)CC1 4135,Cc1cocc1C(=O)NC1CCCC1CC(=O)NCCC1(C)CC1(F)F 4136,CCCS(=O)(=O)CC(=O)N1CCN(C(=O)OCCCOC)C(C)CC1=O 4137,Cc1nc(C(N2CC(OCC(N3CC(C)CC3C)=O)C2)=O)c(C)o1 4138,CC1CC(C(N2CC(NC(c3c(Cl)noc3C)=O)C2)=O)CC(C)C1 4139,N1(C(c2c(C)cc[nH]2)=O)CCC2(CC1)CC2NC(c1cc(I)ccc1C)=O 4140,N1(C(c2ccc(F)nc2)=O)CC2(CCN(Cc3ccc(-n4cccc4)cc3)C2)C1 4141,c1(CC)c(C(N2CCCC(NC(=O)C(C)c3ccsn3)C2)=O)cnn1C(C)(C)C 4142,C(=O)(C(CCC)C(C)C)NCCOC1N(C(CC(=O)OCC#C)=O)CCC1 4143,N1(C(C2ON=C(CC)C2)=O)CC2CC1CC2NC(=O)Cn1ccnc1 4144,c1(C(N(C)CC2(NC(C3N(C(C)C)CCC3)=O)CC2)=O)nc2ccccc2s1 4145,C12(C(=O)NC3C(C(C)C)C3)CCCC1CCN2C(=O)CCCN(C)C 4146,c1(C(=O)NC2CONC2=O)ccc2c(C(N3CCC(Br)C3)=O)n[nH]c2c1 4147,C1(CNC(Cc2c(C)scc2)=O)CC2CCC1N2C(C1(C(N)=O)CC1)=O 4148,c1(NC(C2CC23CCN(C(=O)Nc2ccccn2)C3)=O)ccnc2c1CCO2 4149,C1(CN(C(=O)CN2CC(C)(C)C2)CC)CCN(C(=O)C(C)CC#N)CC1 4150,C=C=CCCC(=O)NCC1CN(C(=O)C=C(CCC)CCC)C1 4151,Cc1ncc(Br)c(C(N2CCC(NC(=O)C3=CCCCO3)C(O)C2)=O)n1 4152,C1(N=[N+]=[N-])(C(=O)NCCC(CCC)C)CCN(C(=O)CCC(=O)NC)C1 4153,C1(C(=O)NC2CC3CC4C(C3)C24)(CC)CCCN(C(=O)COC2CCC2)C1 4154,C1(NC(C(C)CC(N)=O)=O)CCC2(CC1)CC2NC(C1CC(=O)N(C)C(=O)N1)=O 4155,c1(C(N2CC=CC(NC(=O)CC3CCC(F)(F)CC3)C2)=O)ccc2n[nH]cc2c1 4156,CC1CCC(NC(=O)Cc2cc(O)cc(Br)c2)CN1C(c1cccnc1O)=O 4157,S(=O)(=O)(c1cccc(=NCCc2cnccn2)[nH]1)N(C(C)CC#N)C 4158,C(CCCCCN=[N+]=[N-])NC(CCc1cccc(OC)c1)=O 4159,CC1(C)CN(C(=O)CN2CCOC2=O)CCC1C(N1CCCN(CCO)CC1)=O 4160,N1(C(C(C)CN(C)C(C2CCCCC2O)=O)=O)CCOC2(CCC2)CC1 4161,C1(NC(c2c(C)sc(-c3ccco3)n2)=O)CN(C(C2CCC2C)=O)CC12CCC2 4162,c1(C(=O)NCCCNC(c2nnn(C)c2C(F)(F)F)=O)ccc(C2CC2)nc1O 4163,Cc1cc(C(=O)NC2(CO)CCN(C(C3OCCN(C)C3=O)=O)C2)nnc1C 4164,C1(NC(C2=C(C)CCC2)=O)COC2C(NC(c3cccc(O)n3)=O)COC12 4165,C1(NC(C2(C)CC(C)C2)=O)CN(C(=O)CCc2ccc(F)cc2F)CCC1CO 4166,N1(C(C2(C)CN(C)C(=O)C2)=O)CC2CCC(CNC(C3CCCS3(=O)=O)=O)C2C1 4167,O=C(C1CCCn2ccnc21)N1CCCC1c1ccccc1 4168,Cc1c(CN2CCCC(C(=O)Nc3ncc(Br)nn3)C2)cccc1Cl 4169,c1(C(C)=O)[nH]ccc1C(=O)NCC1(NC(=O)CN2CCC(C)C2)CCC1 4170,C(=O)(C1=CC2(CCOCC2)C1)N1C(CNC(=O)CSCC(F)F)CCC1 4171,c1(CC)ccc(O)c(NC(C2(CNC(=O)C(C)OCCC(C)C)CCC2)=O)c1 4172,C1(C(N2CCN(C(CC3CC(=O)C3)=O)C(CO)C2)=O)CC2C=CCC(C1)C2 4173,N1(C(c2ccc(C(C)O)cc2)=O)CCCCC(NC(C2(n3cnnn3)CC2)=O)C1 4174,C1(CC(=O)N(C2(COC)CCOC2)C2CC2)C(=O)NN=C1C.C12(CCC1)C(=O)N2 4175,c1(CCC)nc(C(=O)N(C2CCN(C(C3(C)CCCO3)=O)C2)CC)cs1 4176,c1(OC)cccc(OCCC(=O)NCCC2COCCN2C(=O)C(F)C(C)C)c1 4177,C1(O)(CCNC(c2cn(C3CCOCC3)nn2)=O)CN(C(C2CCC2(F)F)=O)C1 4178,C(=O)(C1=CS(=O)CCC1)NCC(N)CC(F)(F)F 4179,c1(NC(C2(F)CCN(C(c3ccc(F)c(F)c3)=O)C2)=O)nc2ccc(Cl)cc2[nH]1 4180,n1(CCNC(C=C(CCC)C)=O)cc(CNC(=O)CN(c2cnccn2)C)nn1 4181,c1(C(=O)NC2CC3N(C(C(CC)OC)=O)C(CC3)C2)cc2ccccc2cc1F 4182,c1(SC)ncc(Br)c(C(=O)NCC2CC(F)CN2C(=O)C(c2ccccc2)C)n1 4183,c1(CNC(CSCCOC)=O)ocnc1C(=O)NC(C1CCOC1)CO 4184,C1(CCCNC(c2c(C)c[nH]n2)=O)CCN(C(c2cccnc2C2CC2)=O)CC1 4185,C1(C(=O)NCc2csc(O)n2)(CNC(N2CC(C(=O)NC)C2)=O)CCCO1 4186,C(C(=O)N=S1(=O)CCC2(C1)NC(=O)NC2=O)c1ccc(Nc2c(C)ncnc2)cc1 4187,N1(C(c2c(CC)ncs2)=O)CCC2CCCC12C(=O)N(CC(F)(F)Cl)C 4188,Cn1nccc1C(CNC(=O)Cc1ncco1)NC(=O)C(F)C1CCCC1 4189,c1(C(C(=O)NCCCC)N(CC=C)CC2CC2)ccc2ccccc2c1 4190,c1(OC)ccncc1NC(=O)C=C(C)CNC(=O)Cc1ccncc1Cl 4191,C1(CNC(C=CC=CC)=O)CCCN1C(=O)C(F)n1ccnc1 4192,N1(C(c2nncc(C)c2)=O)CCC(F)(F)C(CNC(C2CC=CCC2)=O)C1 4193,O=C(N=c1[nH]nc(Cl)cc1Br)C1CCCN1C(c1cn2c(Br)cccc2n1)=O 4194,C(=O)(CCC(C)OC)N1C(CNC(CCCOCC)=O)CCC1 4195,CCC(CC)CCCC(=O)NC(COC)C(=O)N(CC(C)COC)C 4196,c1(C(C(=O)NCCCN(C(C(C)(C)OC(C)=O)=O)C)C)ccc(C)cc1 4197,c1(C(C)NC(C)(C)C)ccccc1Br.c12cc(on1)C(C)(C)C1CCCN1C2 4198,C1(C(=O)NCCCOCC)CCCN(C(c2nc(C)sc2C)=O)CC1 4199,C1(CC)CCN(C(c2cc(F)c[nH]2)=O)C1CNC(=O)CCc1nncs1 4200,Cc1ccc(OC(C)C(=O)N2CCC2CNC(=O)CCC=CC(C)C)c(C)c1 4201,C=CC(CC)CC(=O)NC1C2CCN(C(=O)C(c3cscn3)N(C)C)CC12 4202,C(=O)(C(O)CCCNC(c1cccnc1)=O)N1CCC(OC)C1C1CC1 4203,c1(C(N2CC3C(C(=O)NC(C(C)C)C)C3C2)=O)c[nH]c2ccccc12 4204,CCCC(CCC)C(=O)NCC1(NC(C2CCCNC2=O)=O)CC(F)(F)C1 4205,C1(NC(=O)CCc2ccc(O)cc2)COCCN(C(C2CC2C2CCC2)=O)C1 4206,c1(C2(C(=O)NC3CCC(CCNC(c4n(C)nnc4)=O)C3)CC2)ccc(Cl)cc1 4207,c1(C(=O)NC(C)C(C)NC(c2csc(O)n2)=O)ccc(-c2cnnn2C)cc1 4208,C(C(=O)NCc1nccs1)(C(C)(C)C)NC(=O)NC1C(c2ccn(C)n2)C1 4209,C=CC1OCCC1C(N1CCCCC1CC(=O)NCC1CCC1C(=O)NC)=O 4210,C1(NC(CNC(CNC(C)=O)=O)=O)CCCN(C(=O)CC2CN(C)CC2O)C1 4211,N1(C(C(=O)NC(C)C)=O)CCC2CCC(NC(=O)CCCC(F)(F)F)C12 4212,C1(C(=O)NC(CC)(CNC(=O)C(C)CC2CCCO2)CC)CC2(COC(=O)N2)C1 4213,c1(-c2ccc(C(=O)NCCCOC)c(C)n2)cccc2nn(C)c(C)c12 4214,C1(NC(COCCCC)=O)CCCC1(C)CN(C(=O)CC1CC1C(F)(F)F)C 4215,C1(NC(=O)CCn2ccnc2)C2CCN(C(=O)C(F)(F)c3nccs3)CC12 4216,C1(CNC(CC(c2cccc(C(F)(F)F)c2)C)=O)CC(F)(F)CO1 4217,c1(C(N2CC(CO)C(CO)C2)C(=O)NC(CC)(C)C)nc2ccc(OC)cc2s1 4218,Cc1cc(C(=O)NC2(c3cn(-c4ccc(Br)cc4F)nn3)CCC2)cc(O)c1 4219,CC1CCn2cc(C(=O)NCC(C)(C)NC(C34CC(C)C3C4)=O)nc2C1 4220,c1(NC(=O)N(C2CCOC2C(F)(F)F)Cc2cccc(F)c2)cccc(Br)c1 4221,Cc1ccc(CC(N2CCC(N(C(=O)CC(=O)NC3CC3)C)C2)=O)cc1Cl 4222,N1(C(C(C)OC)=O)CCC(F)(C(=O)NCCc2cnn(C)c2C)C1 4223,S(=O)(=O)(c1cncc(C(=O)O)c1)NCC1(C(=O)O)CC(OC)(OC)C1 4224,c1(C(=O)NC2(C(N3C(CC)CCC3)=O)CC2C)cnccc1C#N 4225,C(Cc1cnc[nH]1)(C(=O)NOC1CCC(O)C1O)NC(C1CN2CCC1C2)=O 4226,c1(C(=O)NCC(C)(C)OCCNC(C(C(CC)O)C)=O)c([N+](=O)[O-])c(C)nn1C 4227,C1(Cn2c(N3CCN(C(C)=O)CC3)nnc2CC2CCOC2)CCC(F)(F)CC1 4228,CC1(C)CCN(C(=O)C(c2ccc(F)cc2)(C)F)C(C(=O)O)C1 4229,c1(C(=O)NCCCOCCNC(=O)Cn2cncn2)coc2c1C(O)CCC2 4230,c1(CCC)cc(C(=O)N(C2CCC(NC(C3CC4CC3C4)=O)C2)C)cc(O)n1 4231,N1(C(Cc2c(C)nccc2)=O)C(C(=O)NCC2(C)CSC2)C2CC(O)C1C2 4232,N1(C(C(CC2CC2)OC)=O)CCC(C2CCN(C(=O)C(C)(C)CF)C2)CC1 4233,CCC(C(=O)NC(C)CCCNC(=O)C(=O)N(C)C)C(C)(C)CC 4234,c1(C(=O)NC2COCC2NC(C2CC2F)=O)cc2occc2[nH]1 4235,c1(-c2ccc(CN(C(C)(C)C)CC)cc2)ccc(F)c(C)c1 4236,S(=O)(=O)(c1ccc(Br)cc1NCC(C(F)F)n1cccn1)NC(C)(C)COCCO 4237,Cc1ccc(C=C(C#N)C(=O)N2CC(NC(=O)C(C)N(CC(C)C)CC#N)C2)cc1 4238,C(CC(C(=O)N1OC2CCC1CC2)NC(c1cncnc1)=O)=CC 4239,Cc1nc2cc(C(N3CC4CC3C4NC(C3COCCN3C)=O)=O)cnc2[nH]1 4240,c1(-c2ccc(C)o2)ccc(C(N2CCCC2(C)C(=O)NCCC(C)CO)=O)cc1 4241,N1(C(C(C)Cc2ccccn2)=O)CCN(C(c2cc(Cl)ccc2N)=O)C(C)C1 4242,C1(N(C(C2N(C)CCN(C)C2)=O)Cc2nccs2)CC12CCN(C(=O)CO)CC2 4243,CC(CC(F)F)C(=O)N1C(C(=O)N(CC(=O)NC(C)(C)C)C)CCC1C 4244,N1(C(C(CC)(C)O)=O)CCN(C(=O)CCCCCNC(C)=O)CC(C)(C)C1 4245,c1(C(=O)NCC2CCN(C(C3(OC)CC3)=O)C2)cn2ccccc2n1 4246,N1(C(C)C(c2ccc(OC(F)F)cc2)=O)CCC2(CC(C(=O)N(C)C)=NO2)C1 4247,c1(C(=O)NCC(CNC(CN(C(=O)OC)C)=O)C(F)(F)F)cc(C)c(F)c(C)c1 4248,C1(C(=O)NC2C(C(=O)NCC3(OCC)CC3)CCCC2)C2CCC(C2)C1C 4249,c1(CCNC(C(=O)Nc2c(C(C)(C)C)cccc2)=O)nc2ccccc2s1 4250,C(C(CC(=O)N1CCC(NC(C2(C)CCCCCCC2)=O)C1C)C(F)F)N(C)C 4251,c1(CC(=O)OCCCCC(C)=O)c[nH]c2ccc(F)cc12 4252,S(=O)(=O)(c1cc(F)ccc1C)Nc1c(C)cc(F)c(-c2ccncc2)c1 4253,C1(NC(CC2COCC(C)O2)=O)CC=C(C(=O)NCCC(C)N(C)C)C1 4254,c1(OC)ccc(C(Cc2ccc(Cl)cc2)Nc2ccc(C)nc2CO)cc1OC 4255,c1(-c2cn(C(C)C(N3CCC(OCCO)C3)=O)nn2)c(Cl)cncc1Cl 4256,c1(C(=O)NC2CN(C(C3CC(=O)N(C4CC4)C3)=O)C2)cc2c(s1)CCOC2 4257,C(C)(C)(CC(F)C(=O)NC1CC(CO)C2CC12)NC(C(n1c(C)ccn1)C)=O 4258,c1(C(=O)NCCCCCNC(Cc2nc(C)[nH]n2)=O)ncnc2sccc12 4259,S(=O)(=O)(c1ccc(N2CCC2)c2cnccc12)N1CC(C)(CC)OC(C)(C)C1 4260,N1(C(c2ccnn2CCF)=O)CCCC(CNC(C2CC(O)C2)=O)C1 4261,Cc1ccc(C#N)c(NC(=O)CC2CN(Cc3ccc4c[nH]nc4c3)CCO2)c1 4262,CCC(CC(F)(F)F)C(=O)NC1(C)CC(NC(c2cc(Br)cn2C)=O)C1 4263,N(C(=NCCCCl)NC1CCN(C2CCCC2)C1)Cc1c(C)nns1 4264,C(C)(C(=O)NC1CCC(n2cc(-c3ccc(C)nc3)nn2)CC1)(C(C)C)OC 4265,c1(C(N2CCC(NC(C(CC(C)C)NC(N)=O)=O)C2)=O)csc(N=S(C)(C)=O)n1 4266,C1(C(=O)NC(c2occ(C(N(C3CCOC3)CC)=O)n2)C)CC(C)N(C)C1 4267,C1(CNC(CNC(c2ccc(SC)s2)=O)=O)CCCN(C)C1=O 4268,c1(COCC(N2CC(O)(C(C)NC(CC=CC=C)=O)C2)=O)ccccc1Cl 4269,c1(OC)cccc(NC(c2cc(C)cs2)c2nnnn2-c2ccccc2C)c1 4270,C(=O)(CCCCCS(N)(=O)=O)N1CCC(C)C(NC(=O)CCCC(=O)C2CC2)C1 4271,C(=O)(CC1=NNC(=O)C1)NC1CN(C(c2n(C)cnc2)=O)CC(O)C1 4272,Cc1cccc(F)c1C(N1CCN(C(=O)C(c2ccc(Cl)cc2)(F)F)CC1C)=O 4273,N1(C(C(COC)C)=O)CCCC12CCN(C(C1CCC(=O)C1)=O)CC2 4274,c1(CC(C(=O)NC2(CC)CCOC2)C)ccc(OC)c(OC)c1 4275,c1(C(=O)NC2C(CO)CCN(C(C3NC(=O)OC3)=O)C2)cnn2c1OCCC2 4276,[N-]=[N+]=NC1CCC2(C(=O)NC3CC(F)C3)CC12 4277,N1(C(C2C(C=C)C2)=O)CCC(C2(NC(=O)Cc3cc(C(F)(F)F)n[nH]3)CC2)CC1 4278,c1(CS(N2CC(F)(C(=O)O)C2)(=O)=O)nc(Br)ccc1N 4279,C1(NC(c2ccc(CC)o2)=O)CCN(C(=O)C(O)Cn2cncn2)C1(C)C 4280,c1(C(=O)NCC(C23CCC(CC2)C3)NC(CC(=C)C)=O)ccc2ncncc2c1 4281,N1(C(CC)=O)CC2CC2(CNC(=O)C(N2CCNC2=O)C)C1 4282,N1(c2cc(C)nc(Cl)n2)CC2CC1CCC2NC(=O)CC(C)n1ccnc1 4283,CC1CC(C(=O)N(C(C)CNC(C2CCC(C(C)(C)C)O2)=O)C)CC(C)C1 4284,C1(C(=O)NC(CC=C)CNC(c2csc(NC=O)n2)=O)CCc2ccccc2O1 4285,C12(CNC(CC=C)=O)COCCN1C(=O)CN(C(C1CC1C)=O)C2 4286,N1(C(c2cncc(C#N)c2)=O)CCCC(C2(NC(=O)CCC3CCOC3)CC2)C1 4287,C1(C(N2CC(n3ncc(NC(C=C(C)C)=O)c3)C2)=O)COCCN1C 4288,N1(C(C=COCC)=O)CCSC(C(N2CCC(c3cncc(C)c3)CC2)=O)C1 4289,n1(CC)nnc(C(=O)NC(C2CN(C(C3(C)CCCOC3)=O)C2)C)c1C 4290,N1(C(C=CC(=O)N(C)C)=O)CCC(C)(C)C1CC(=O)NCC=CCO 4291,c1(C(N2CCC(COC)(NC(=O)CCCF)C2)=O)cc2c(cn1)OCCC2 4292,c1(C(=O)NCC(C)(C2CC2)NC(C(C)OCC#C)=O)cncc(F)c1C(F)(F)F 4293,CC1CN(C(C2CCC3(CCC3)O2)=O)CCN(C(=O)CCc2cn[nH]c2)C1 4294,C(=O)(C(CC(C)(C)C)NC(=O)C1=C(C)OCCC1)N1CC(CCC)C(OC)C1 4295,c1(C(C(=O)NC(C(C)(C)NC(c2c(C)con2)=O)C)C)cc(F)cc(F)c1 4296,S(=O)(=O)(c1ccc(Cl)cc1)N1C(C(=O)NC(C(C)C)CCO)C2CCC1C2 4297,c1(C(N2C(CNC(CSCCCC)=O)C(CC)CC2)=O)cc(F)cnc1O 4298,C1(C(C)NC(=O)CCCc2cncs2)CCCCN1C(=O)Cn1cnc(C(N)=O)n1 4299,CC1(C)C(NC(c2cc(Cl)ccc2Cl)=O)CC1N=c1ccnc(Cl)[nH]1 4300,C1(CNC(C(C)NC(c2ccco2)=O)=O)CC12CCN(C(=O)C=C1CCC1)CC2 4301,CCCC(O)C(=O)N(CC)CC1CCCN(C(=O)C(C)CC2CCCCC2)C1 4302,CCCCC(O)CNC(=O)CC1COCCN1C(=O)CC1CCN(C)C1=O 4303,N1(C(C2(C)C(C(=O)OC)C2)=O)CCC2(C1)CN(C(=O)C(C)(C)CC(C)=O)CCO2 4304,C1(NC(C(C)(C2CCC2)NC(C=CCC)=O)=O)CCCCNC1=O 4305,C(=O)(CCP(C)(C)=O)N(C(C)C)CCNC(C1(c2cccc(Cl)n2)CC1)=O 4306,N1(C(c2c(C)[nH]nc2Br)=O)CCN(C(=O)CCC2CCCOC2)C(CO)C1 4307,c1(C(=O)NCC(C)(C)O)cc(F)ncc1NC(C1(CCCCO)CC1)=O 4308,CC1(CNC(=O)C(C2(O)CCCC2)F)CCN(C(C2C3CCCC23)=O)C1 4309,N1(C(C(=O)NCC(CC)NC(=O)CCOC(C)C)C)CCCCC1 4310,c1(C(=O)NCC2N(C(c3ccc(OC)nc3)=O)CC(F)C2)c(C)nn(CC)c1Cl 4311,N1(C(C2CNC(=O)N2)=O)CC2CCC1C1CN(c3c(Br)cncc3[N+](=O)[O-])CC21 4312,c1(OC)cc(C)ccc1C(N1CC2CC1C2NC(c1ccnnc1)=O)=O 4313,c1(C(N(CCNC(c2ccc(O)c(O)c2)=O)CC)=O)cc2cc(C)ccc2s1 4314,CC1COCC(CC(=O)N(C)CCNC(=O)C(c2cccc(Cl)n2)(F)F)O1 4315,C1(C(=O)NCCCC(C)NC(CC2(C(=C)F)CCC2)=O)CCC2(CC1)CC(=O)C2 4316,c1(OC)cc(C(N2CCCCC2CN(C(=O)C(O)COC)C)=O)ccc1F 4317,c1(C(=O)NCC2CC(OC)CN2C(=O)CN(C)C(C)C)ccc2c(c1)N(C)CC2 4318,C(CCCCCS(=O)(=O)CCO)NC(=O)NC1CCC=CO1 4319,c1(C(N2CCN(C(C(C)CC3CC3)=O)CC2)=O)cccc2c1OC(C)C2 4320,n1(CC(N2CC(CCNC(c3cnccc3Cl)=O)OCC2)=O)cnc([N+](=O)[O-])c1 4321,c1(CN(C)C(C2CCN2C(C2CCCC2O)=O)=O)nccn1C 4322,c1(C(N(C)CC2CN(C(c3cn(CC)nn3)=O)C2)=O)ccncc1OC 4323,Cc1ccc(C(=O)NCCC2(NC(c3cccnc3N)=O)CCC2)c(Cl)c1 4324,c1(C(N(CC(C)NC(CSCCOC)=O)CC)=O)cnn(-c2ccncc2)c1 4325,Cc1n[nH]cc1C(N1CCC1CNC(c1c[nH]nc1-c1ccsc1)=O)=O 4326,Cc1nc(NCCN2CCCCCC2=O)cc(NC(C)C(C2CCCCC2)O)n1 4327,C(CCCCn1cc(CO)nn1)NC(=O)NC1CCN(c2ccccc2)C1 4328,N1(C(C(C)=CC)=O)CC2CCCCC2(CNC(=O)COc2cc(F)ccc2F)C1 4329,N1(C(c2nc(CC)oc2C)=O)CC2CC1CN(C(C1(C(N)=O)CCC1)=O)C2 4330,C(=O)(CC(c1ccccc1)C1CC1)NCCC(C)N(C(CCNC(C)=O)=O)C 4331,N1(C(CCN2CCC(C)CC2)=O)CCC(NC(c2ccc(Cl)s2)=O)C(CO)C1 4332,N1(C(C2CCC(N(C)C)CC2)=O)CCCC2(NC(=O)C3=CCOCC3)CC2C1 4333,c1(CNC2CC(C(N3CCC(F)C3)=O)C2)cnn(-c2ccccc2)c1 4334,N1(C(c2cc(C)c(F)cc2)=O)CC2CCN(Cc3ccc(CO)o3)CC2C1 4335,CCC(C)CCC(O)CC(=O)NCC1(NC(C2CCCN2CC(C)C)=O)CCC1 4336,C#Cc1cc(C(C(=O)NCC2CCOC2)N(CCC#N)CC2CC2)cc(Br)c1 4337,N1(C(c2c(CC)[nH]nc2Cl)=O)CCC(NC(=O)Cn2cc(N)cn2)C(C)(C)C1 4338,C(C(CC1CC1)C(=O)N1CC(O)C(F)C1)NC(c1ccn(COC)n1)=O 4339,c1(CCN(C)C)ccc(C(=O)NCC(CO)NC(c2occc2C2CC2)=O)cc1 4340,C1(OC)CCCC(C(=O)NC(CNC(C2CCOCC2)=O)C(C)C)C1 4341,c1(C(N2CCC(N(C(C3CCC4CCC3O4)=O)CCO)C2)=O)c[nH]cc(F)c1=O 4342,CCCCCC=CC=CC(=O)NCCOCCNC(c1cc(C)no1)=O 4343,N1(C(C(C)(CO)OC)=O)CCC2(CC1)COC(CNC(c1coc(C)c1)=O)C2 4344,Cc1ccc(C(N2CCC(CC(=O)NCCn3ccnc3C)C2(C)C)=O)cc1C#N 4345,C1(NC(=O)C=Cc2ccc(C3CC3C)o2)CN(C(=O)C(Cl)=CCl)CC2(CCC2)C1 4346,C(CC(C)(C)C(=O)NC(C)CC(C)NC(C1(C)SCCCS1)=O)OC 4347,Cc1ccc(F)c(NC(=O)C(=O)NC2CC(c3ccccc3)C2C)c1 4348,CC1CCC(C(=O)NCc2cscn2)N(C(C2CC2C(=O)OC)=O)C1 4349,CCCC(C(=O)OC)C(=O)NC1CC(CNC(c2cc(Cl)ns2)=O)C1 4350,Cc1nn(C)cc1CC(=O)NCC1COCCN1C(C1CC(CC(F)(F)F)C1)=O 4351,C(=O)(C(C)(C)Cn1cccn1)NCC1CN(C(C(C)c2ccsc2)=O)C1 4352,C1(NC(C2N(C(CC3CC(SCC)C3)=O)CC2)=O)CC(CO)N(C)C1 4353,C1(C(=O)NC2CCN(C)C(=O)C2)CC12CCN(C(=O)CC1C=CCC1)CC2 4354,c1(CC)ccc(C(=O)NC2(C(=O)ONCC(=O)NC(C(C)NC(C)=O)C)CC2)cn1 4355,C(=O)(CCCN(C(=O)C(C)NC(c1ccoc1C)=O)C)NC 4356,N1(C(C2CC(=C)C2)=O)CCC2(CC1)CN(C(c1n[nH]c(C)c1[N+](=O)[O-])=O)CCO2 4357,C(=O)(C(C)(C)S(C)(=O)=O)NC(C(C)NC(c1cc2c(s1)CCC2)=O)C 4358,C#CC1(O)CCCC(NCc2ccnc(N3CCOCC3)c2)C1 4359,c1(C(=O)NCC(F)CNC(c2coc(Cl)n2)=O)cccc(N2CCOC2=O)c1 4360,c1(C(=O)NCCN2CCN(C(C3(C#N)CC(C)C3)=O)CC2)n[nH]c2ccccc12 4361,c1(NC(=O)CC2CCCN2Cc2cccnc2)cc(Cl)c(Cl)cc1F 4362,c1(C2C(C(N(C3CCN(C(c4sccc4Cl)=O)C3)CC)=O)C2)c(C)n[nH]c1C 4363,c1(COC)ccc(C(=O)NCC2CC(C(=O)N(C)Cc3ncn(C)n3)C2)o1 4364,Cc1c(C(=O)NC2CN(C(=O)CCc3nc(=N)[nH][nH]3)C3CC23)c(C(F)F)nn1C 4365,c1(NC2C(CNC(CN(C)C(N)=O)=O)CCCC2)ccc(C#N)nc1 4366,C1(NC(C(CCOC)C)=O)CN(C(=O)C(=Cc2ccccc2)C#N)CC1(C)C 4367,CC1(C)CC=CCN(C(C23COCC2CN(C(C24CSCC2C4)=O)C3)=O)C1 4368,c1(C(=O)NC(C(C)NC(c2c(SC)n(C)nc2)=O)C)c(C)ccc(C)c1C 4369,CC1CCC(C2CCC2)CN1c1nnc(-c2ncc(Cl)cc2Cl)n1CC1CC1 4370,C1(NC(c2c[nH]cc2Br)=O)CCN(C(=O)C=C2CCSCC2)C12CCCC2 4371,C(CC(C(F)F)c1ccccc1)NC(c1nnnn1-c1ccccc1)CCC 4372,c1(COC)nc(Cl)cc(=NCC(C(C)(C)C)NC(C2CC3(CC(C)=NO3)C2)=O)[nH]1 4373,C(CCC(C)C(=O)NCC12CCC(CC1)N2C(=O)CCC1OCCO1)OC 4374,C1(C(=O)NC2CC2C(=O)NCc2cccc(CO)n2)(CC)CCCCC1 4375,c1(-n2c(N(C3CC4(CNC4)C3)C(C3SCC(=O)C3)=O)ccn2)ccc(F)c(Cl)c1 4376,c1(N2C(=O)CN(CC)C2)ccc(OC(C2CC23CC(CNC(=O)NC)C3)=O)cc1C 4377,c1(CC(=O)NC2CC(C(=O)Nc3c(C(=O)OCC)ccs3)C2)ccnc(Br)c1 4378,C(=O)(CCC(CF)CF)NC(C(CC)C)C(=O)N(CC(=O)NC(C)(C)C)C 4379,c1(C(C(=O)NCC(CNC(Cc2c(C)occ2)=O)O)F)ccccc1F 4380,C(CC(C)(C)C(=O)NC1CCN(C(c2scnc2Cl)=O)CC1F)SC 4381,c1(CCCC=C)cn(C(COCC)C(=O)N2CCC(c3ccco3)C2)nn1 4382,c1(C(N2CC(O)CC(NC(c3cnc(O)cc3O)=O)C2)=O)c(Cl)ccc(O)c1Cl 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4419,C1(COC)(NC(C2Cc3nnsc3S2)=O)CCC(C)(C)CC1 4420,Cc1ccc(SCCCN(C(C(N2CCOC(C(F)(F)F)C2)=O)C)C(C)C)cc1 4421,c1(C(=O)NCC(CNC(CC2(C)CCCCC2)=O)F)nccc2c1CNC2=O 4422,C(=O)(NNC(=O)C(C)(C)CCCCNC(=O)C(F)(F)CC1CC1)C1CC(C)C1O 4423,c1(N2C(C)CC(NC(C3(C4CCC4)CC3)=O)C2)ncnc2[nH]ccc12 4424,C1(NC(C(C2CCCCC2)OC)=O)CN(C(c2nccnc2C)=O)CCC1F 4425,C1(C(=O)NC(C(C)(C)C)CNC(=O)CNC(=O)C2CC2)CCC2C(CC1)C2(F)F 4426,Cc1ccc2c(Br)cnc(N3CCNC(=O)C3c3cnn(C)c3)c2c1 4427,CN=c1nc(C(N2CCC(CSC3COCCN3)CC2)=O)cc[nH]1 4428,c1(OCC)ccc(CN2CCC(NC(c3cc(Cl)ccc3I)=O)CC2)cc1OC 4429,N1(C(CNC(C(C)OC)=O)=O)CCC(COCC(F)(F)C(F)F)C(C)C1 4430,N1(C(C2CC(=O)OC2)=O)CCN(C(C2(CF)CC(F)(F)C2)=O)CC1CC(F)(F)F 4431,CCCC(CC)CCC(=O)NC1C=CCN(C(=O)C(C)(C)OC(C)=O)C1 4432,C1(C(=O)NCCCc2n(CC)ncc2)C2CCC1N(CC)C2 4433,c1(C(=O)NCC2C(NC(C)=O)CC2)cc(C)c2n[nH]cc2c1 4434,Cn1c(C(N2CCN(C(c3cccc(CO)n3)=O)CC2)=O)cnc1O 4435,c1(C(C)C)nn(C)cc1C(=O)NCC1CN(C(c2csc(C3CC3)n2)=O)CCO1 4436,C(=O)(C(O)CC(C)(C)C)N(C1CCN(C(=O)Cc2c(F)cccc2Cl)CC1)C 4437,S(=O)(=O)(c1ccc(Br)s1)N1C(CC(=O)N(C2CCC2)CCO)COCC1 4438,c1(CC(N2CCC(NC(=O)CC3CC4CC4C3)C2)=O)cccc(Br)c1Cl 4439,N1(C(c2c(C)cccc2)=O)CC(NC(=O)CC2NC(=O)NC2=O)CC2(CCC2)C1 4440,c1(C(=O)NCC2C(CNC(C3(C(C)(C)O)CC3)=O)C2)ccnc2[nH]c(O)nc12 4441,n1(CC(=O)NCC(CNC(c2c(CC)nc[nH]2)=O)CO)cc(Cl)c(C)n1 4442,N1(CC(N2C(C3(CNC(C(C)NC(CC)=O)=O)CC3)CCC2)=O)CCNC(=O)C1 4443,C1(NC(Cc2nnc(C)s2)=O)CCC2CN(C(C3CCS(=O)(=O)C3)=O)CCC2C1 4444,c1(C2(C(N3CC(CCNC(CC(C)OC)=O)C3)=O)CC2)ccc(Cl)c(F)c1 4445,N1(C(CC(CC)C)=O)CC2CN(C(=O)Cc3ccc(OC)c(O)c3)CC2C1 4446,c1(NC(c2cnc(C)s2)C)ncccc1S(=O)(=O)NCC1CCC1 4447,c1(C(C)NC(c2scc(CNC(CC3(OC)CCC3)=O)c2)=O)ncccc1F 4448,N1(C(C2C(C)CCC2)=O)CCC2(C1)CN(C(c1ccc3nccn3c1)=O)CCO2 4449,N1(C(C(C)OC)=O)CCC(C(C)(C)NC(C2CC2C)=O)CC1 4450,C1(C(N(CCN(C)C)C)=O)CCN(C(=O)NC2CCCCN2)CC1 4451,C12(NC(CN(CCOC)C)=O)CCC(CC1NC(=O)Cc1sc(C)nc1C)C2 4452,C(=O)(CCC(C)=O)NC(c1cnn(C)c1)C(N1CC(OC)(CO)C1)=O 4453,CC1(C#N)CC(c2nnnn2Cc2ccccc2)(NCCCC2CC2)C1 4454,c1(C(N2CC(NC(C3ON=C(C)C3C)=O)C(C)C2)=O)ccc(=O)n(C)c1 4455,CC1(C)CCC(N=[N+]=[N-])CN1C(c1nc(Cl)ccc1Cl)C(=O)NC(F)(F)F 4456,N1(C(C(n2cc(-c3cccc(N)c3)nn2)C)=O)CCN(C(C)(C)C)C(C2CC2)C1 4457,Cc1cc(NCC2CCCO2)nc(N(C)CCn2cncn2)n1 4458,c1(C(=O)NCC(CC)NC(C(CC=C)C)=O)ccc(Br)c(C(=O)OC)c1 4459,N1(CCS(=O)(=O)N2CCCCC2)CCOC(c2cccc(Br)c2)C1 4460,C(=O)(C(CC)C(=O)OC)NCCCC(=O)NC1C(CC=C)CCCC1 4461,N1(C(c2cc(CC)[nH]n2)=O)CCN(C(=O)C(O)CC(C)C)CC1C1CCCC1 4462,Brc1cccc2c1C(NC(c1nnnn1C1CCOCC1)C1CCCC1)CC2 4463,C1(NC(c2cnc(Cl)[nH]2)=O)CCN(C(c2nccnc2C(F)F)=O)CC1F 4464,c1(NC(=O)NCc2ccc(N3CCS(=O)(=O)CC3)nc2)cc(I)c(O)c(I)c1 4465,C1(C(=O)NC(CCC=C)C)CCC(NC(=O)C(O)CN2CCCC2)CC1 4466,N1(C(CN(C(c2nn(C)cc2Cl)=O)CC)=O)CCC(CO)C(O)C1 4467,n1(CC(=O)N(C)CC2CCCN(C(c3cc[nH]c(=N)c3)=O)C2)nc(Cl)ccc1=O 4468,N1(C(c2c(C#N)csc2)=O)CC2CCCC1CN(C(=O)CNC(C1CCC1)=O)C2 4469,C(CCN=c1ccnc(N2CCCC(C)(F)C2)[nH]1)N1CCN(C(COC)=O)CC1 4470,N1(C(Cc2cccc(NC(=O)OC(C)(C)C)c2)=O)CCC2CCOCC2C1 4471,CCS(=O)(=O)CC(=O)N1CC(C)CCC1C(=O)NCCC1CCCC1O 4472,C1(CNC(Cc2c(C)con2)=O)CCCCC1NC(=O)C(=C1CCCCC1)F 4473,c1(C(C(N2CCC(N(CC#C)C(c3[nH]cc(C)c3C)=O)C2)=O)=O)ccc(F)cc1F 4474,N1(C(C2(C(C)(C)C)CCCC2)=O)CCC(C)(CNC(c2cc(CCO)on2)=O)C1 4475,C1(C(N2CCC(OC)(CNC(c3cncc(CO)c3)=O)C2)=O)CC(=O)NC(=O)N1 4476,CC1(C)CCC(CC(=O)NCC(=C2CN(C(=O)Cn3cnnc3)C2)F)OC1 4477,Cc1cc(CNCCC2CCOC2(C)C)nc(Cl)c1Br 4478,N(C)(S(=O)(=O)N1CCN(CC(=O)NCCOC2CC2(F)F)CC1)CC 4479,CCC(CNC(=O)C=Cc1ccccc1C)(CC)C(=O)N1CCC(N(C)C)C1 4480,N1(C(c2cnc(COC)s2)=O)CCCC(NC(C2CCC(C(N)=O)CC2)=O)C1 4481,C(CCCC(C)(C)C(=O)NNC(=O)C12CCCC1C2(F)F)NC(CC)=O 4482,c1(C(=O)OC)[nH]c(=NC(C)Cc2c(Cl)cccc2Cl)[nH]c2ncnc1-2 4483,C(=O)(C(C(C)C)C1CCC1)NCC1(OC)CN(C(c2cnc(O)o2)=O)C1 4484,Cn1ncc(N(C(C2(C)C=CCC2)=O)CC2CC2)n1 4485,c1(CNC(N2CCN(C(=O)Cc3cncnc3)CC2)=O)ccc(F)cc1F 4486,C1(OC)(CNC(C2(F)CCN(C(=O)Cn3nnc(C)n3)C2)=O)CCCCC1 4487,C1(O)(CNC(C(N2CCNC2=O)C)=O)CCCN(C(=O)CCc2cnn[nH]2)CC1 4488,C1(C(=O)NC2CC(F)(CNC(C(C)OCC)=O)C2)CC(C)(C)CC(C)(C)C1 4489,c1(C(=O)NC2CCN(C(CCC=CC)=O)CC2CO)cc2ccccc2nc1O 4490,C(=O)(C(C(=O)NCC(C)(C)CCNC(C1(C)CCNC1=O)=O)OC)OC 4491,c12cnn(c1C)C2.C1(F)(CNC(=O)NC(CCC)C2CC2)CC(CN(C)C)C1 4492,C1(C2CCN(C(c3cc(C)cs3)=O)CC2)(NC(C(CC(C)C)NC(C)=O)=O)CC1 4493,C1(NC(CCCC)Cc2ccccn2)CCc2cc(C#N)ccc2C1 4494,CC(C)C(CCN(C(=O)CC1C(C)C1(F)F)C)NC(c1cnc(S)n1C)=O 4495,c1(OC)cncc(-n2nccn2)n1.C123CC1CN(C2)C(=O)C1CC(C1)NC3=O 4496,C(N=c1nc2c(Br)csc2c[nH]1)C1N(C(C(C)(C)S(C)(=O)=O)=O)CCC1 4497,N1(C(C2OCCN(C)C2)=O)CCC2(CC1)CN(C(c1ncccc1N)=O)CCO2 4498,c1(NC(C)C)ccc(C(=O)NCC2CC2CNC(c2cc(Cl)no2)=O)cn1 4499,O=C(C1CCCc2ccnn21)NCC1CCN1C(c1cnc(O)n(C2CC2)c1=O)=O 4500,N1(C(CN(CC(C)C)C(C2CC(=C)C2)=O)=O)CCOC(C(N)=O)C1 4501,c1(CC(=O)NC2CN(C(CC(C)(C)C#N)=O)CC2(C)C)csc2c(F)cccc12 4502,CC1CCN(C(=O)CN2CC3CCC2C3)CC1CNC(c1cc(Cl)on1)=O 4503,c1(NCCc2c(O)cccn2)[nH]c(=NCCC2CCC2)nc2scnc12 4504,C1(C(=O)OC)CN(C(C2CN(Cc3ncccc3F)CCN2)=O)CCC1O 4505,N1(C(CC2C(=O)NCCC2)=O)CCCC(Cl)(O)CC1 4506,N#Cc1ccc(C(=O)NC2(C(N3CCC3CO)=O)CCSC2)s1 4507,CN1C2(CCN(C(c3cnnc(O)c3)=O)CC2)C(NC(=O)CCCF)CS1(=O)=O 4508,C1(CN(C(Cc2cc(C)sc2)=O)C)COCCN1C(=O)CCCOC(C)=O 4509,C(=O)(C(CCC(C)C)NC(=O)C=Cc1cc[nH]c1)N1C(CC)CCC1 4510,N1(C(C(Cc2cc[nH]n2)NC(c2cnc(Cl)s2)=O)=O)CCC12CCCC2 4511,n1(C(C(N2CC(N(CC(=O)NC(c3onc(C)n3)C)C)C2)=O)C)nc(C)cc1C 4512,CCC(CN=C(NCCn1cnnn1)NC1CCC1)c1cccs1 4513,c1(CN(C(C(=O)OC)C2CC2)C)ncc(C(C)(C)C)o1 4514,N1(C(=O)OC(C)(C)C)CCC=CC1C(=O)OC.C123CC(C1)(C2)CNC3=O 4515,Cn1nc(C(N2CC3CCC(C2)N(S(=O)(=O)CC#N)C3)=O)c2cc(Br)ccc12 4516,c1(CC(=O)NCC23C(CN(C(C(CC#C)O)=O)C2)CC3)ccc(F)cc1[N+](=O)[O-] 4517,C1(C2CCN(CC=C)C2)(NC(N(CC=C)CC=C)=O)CC1.C(=O)(C)OC(C)(C)C 4518,C1(C(N(CC(=O)OC)C2CC2)=O)CCC(O)CC1.c12nncn1CCCC2 4519,C1(CNC(C2C(=C)C2)=O)(COC)CCN(C(c2cc(C)ccc2N)=O)CC1 4520,N1(C(C(C(C)C)O)=O)CCC2(CCN(Cc3nc(-c4ccc(F)cc4)no3)C2)C1 4521,Cc1cnc(C(=O)N(C2CN(C(c3cnnc(O)c3)=O)CC2F)C)c(Br)c1 4522,N1(C(c2c(C)oc(Cl)n2)=O)CCC2(C1)CN(C(C1CC13CCOCC3)=O)C2 4523,N1(C(c2c(SC)cn(C)n2)=O)CC(NC(C2(C(=O)OC)CC2)=O)CC(C)C1 4524,C(=O)(CCCC(=O)C(C)OC(=O)C(F)CC1CC(F)(F)C1)OC 4525,c1(C(=O)NC2CC(CCNC(C(C)P(C)(C)=O)=O)C2)cnc2ncnc(O)c2c1 4526,c1(C(N2C(CN(C(C(CCN(C)C)O)=O)C)CCC2)=O)cc2n(n1)CCO2 4527,N1(C(CC2(C)CCN2C(=O)CCn2cccc2)=O)CCCNC(=O)CC1 4528,CCCC(CCCNC(C1CC1CC)=O)NC(c1ncccc1C(F)F)=O 4529,C1(C2CCN(C(=O)C(F)CC3CCCCC3)CC2)(NC(C(CC)C)=O)CC1 4530,C1(CNC(CNC(=O)OC)=O)CC2COCC2N1C(c1ccn2nccc2c1)=O 4531,C1(N=[N+]=[N-])(C(N(C(C#C)(C)C)C2CC2)=O)CCN(C(=O)CN2CCSCC2)C1 4532,c1(OC)cc(N(C(=O)C(C(C)C)c2ccc(Cl)cc2)C(=O)CC(C)C)ccc1Cl 4533,c1(-c2cc(C(=O)NC3CN(C(c4cnn(CC(F)F)n4)=O)C3)n[nH]2)ccccc1O 4534,C(=O)(CCCC(C)NC(=O)CN1CCCCC1)NCC(C)C#N 4535,N1(C(C(C)CCN(C)C)=O)CCN(C(=O)CC2(C)OCCO2)CC(C)(F)C1 4536,Cc1cc(CC(=O)NCc2nc(C(=O)N(CC(C)O)C)co2)no1 4537,C(=O)(C1=CCCC1P(C)(C)=O)NCC1(O)CN(C(c2c(C(C)C)con2)=O)C1 4538,C1(NC(CCCOCC)=O)CCCN(C(=O)CCC(C)(C)F)CC1F 4539,CC(N=c1[nH]c(NC2C3COCC23)nc2c1SCC2)C1CCC1 4540,CC(C)C(C(=O)NC(C)Cc1ccncc1)C(C)NC(C1CC(=O)C1)=O 4541,C(=O)(CCN(OC)C(=O)C(C)N(C(=O)C(C)C#N)C1CC1)OC 4542,N1(C(CC#N)=O)CCC2(NC(c3ccc(-c4ccon4)cc3)=O)CCCC12 4543,CC1(C)OC(=O)CC1C(=O)NC1CC=CCC1C(=O)NCCc1cccs1 4544,Cc1ccsc1CC(=O)N(C(c1ccccc1)CNC(C1(CC2CC2)CC1)=O)C 4545,c1(-c2c(C)c(O)ccc2)ccc2ccnc(NS(=O)(=O)c3cn[nH]c3)c2c1 4546,c1(C(=O)NCC2C(CNC(c3c(C#N)nc[nH]3)=O)C2)cc2ccccc2o1 4547,n1(CC(=O)NCCCCNC(C2COCCO2)=O)nc2n(c(=O)c1=O)CCC2 4548,C(=O)(CCCCCN(C)C(c1cn(C2CC2)nn1)=O)NCC(CCCC)O 4549,C1(NC(C(c2cncc(F)c2)C)=O)C2CC1CN(C(c1ccc([N+](=O)[O-])[nH]1)=O)C2 4550,N1(C(CC(C)C)=O)CCC(CNC(=O)C(O)CN2CCOCC2)C1(C)C 4551,c1(CC(C)OC)nc(-c2ccc(C3CC3(F)F)cc2)n(C2CCN(C)CC2)n1 4552,N1(C(CC(C)(O)CC(=O)O)=O)Cc2ccc(O)cc2CC1C(=O)NCCC(N)=O 4553,C=CCC(C)C(=O)NC1CCCC(CNC(C2CCN(C(N)=O)CC2)=O)C1 4554,C(N=C(NCC(F)F)N(C)Cc1ccc(Br)cc1)C1(C(=O)OC)CCCO1 4555,c1(Cn2cc(CC3CCCN(C(CC4(C)CC4)=O)C3)nn2)cc(Cl)ncc1Cl 4556,C1(C)(NC(c2nc(C)sc2)=O)CCCCC1C(=O)NCCc1cscn1 4557,CCC(O)CC(=O)NC(c1cccc(Cl)c1)CNC(c1cnn(CC)c1)=O 4558,C(CC(=O)N1CCC(C(=O)NC(CO)C(C)O)O1)OCC#C 4559,N1(C(c2cnn(C(C)C)c2Br)=O)CCOCC(CNC(=O)C(O)C(C)(C)C)C1 4560,N1(CCCCCNC(C2CC23CC3)=O)CCN(C(=O)CC2COCC2O)CC1 4561,C12(C(=O)NCCC3CC(C(=O)NC(C(=O)OC)(C)C)C3)CCCC1C2(F)F 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4635,C=C(CNC(C1CC(NC(=O)C=Cc2cncs2)CCO1)=O)C(F)(F)F 4636,c1(C(N2CCC(CC)C2C(=O)N(C(C)CCC(C)C)C)=O)n[nH]c2ccccc12 4637,N1(C(C(=O)NC)=O)CC(CNC(c2cc(C)c(-c3ccccc3)s2)=O)C(O)C1 4638,c1(CCC)cc(C(=O)NCCC2CN(C(c3occc3F)=O)CCO2)cc(O)n1 4639,C1(CNC(C2CCOC2)=O)CN(C(=O)CSc2ccccc2)CC1CC(F)(F)F 4640,N1(C(c2cc(CC)n(C)n2)=O)CC2CC1CC2NC(=O)C1=CCCC1 4641,c1(C(=O)NC2CCN(CCNC(C(CC)(C)O)=O)CC2)cc(C)cc(O)c1 4642,C(=O)(C1=CCCC1)NC(C1CN(C(C23CCCCC2C3)=O)C1)C 4643,c1(C(=O)NCC(CCC)C(=O)N2CCC2CN=[N+]=[N-])cc2cccnn2c1 4644,C1(=CC(=O)NCC(CN(C(C(C)(C)OC(C)C)=O)C)O)C2CC3CC(C2)CC1C3 4645,N1(C(c2cccc(CC)c2)C(=O)NC)CCCN(C(C2CCCSC2)=O)CC1 4646,C1(CC)(CC)CN(c2cc(NCC(C)(C)CN3CCCC3)nc(C)n2)CCS1=O 4647,C12(NC(c3cc4sccc4[nH]3)=O)CCN(C(=O)C3=CCCSC3)CC1C2 4648,C1(C(=O)NC(C2CC(NC(=O)C(N3C(=O)CCC3=O)C)C2)C)CC(=O)C1(C)C 4649,N1(C(C(C)=CC(C)(C)C)=O)CC=C(CC(=O)N2CCCN(C)CC2C)CC1 4650,CCS(=O)(=O)C=CC(=O)N(C(C)CNC(c1cccn(CC(C)C)c1=O)=O)C 4651,C1(CNC(C)CCc2ccc(C(F)(F)F)cc2)CC(C)(C)CCN1 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4687,c1(C(=O)NC2CN(C(c3cc(C(C)=O)[nH]n3)=O)C(C)C2)ccc(N)cc1Cl 4688,C1(F)(C(N(CCNC(C(C)C(=O)N(C)C)=O)CCOC(C)(C)C)=O)CCS(=O)(=O)C1 4689,C(=O)(CC(C)C(=O)NCC1CC(O)CN1C(=O)Cc1ccnc(C(F)(F)F)c1)OC 4690,N1(CC(N2CCN(Cc3ccc(C)cc3)CC2)=O)CCCC2(CCCCO2)CC1 4691,CC1CCC(C(=O)NOC2CCC2)CN1C(c1cscn1)=O.CO 4692,c1(C(N)=O)cccnc1CNC(C1CCN(c2ccccc2F)C1=O)=O 4693,CC(C)P(=O)(CC(=O)NC1CC2CCC1(NC(=O)CCn1ccnc1)C2)C(C)C 4694,n1(C(CC(N2CCC(N(C(CC)=O)CC)C2)=O)C)nc(C)cc1C 4695,c1(C(N(C(CC)C(=O)OC)CC)=O)cc2sc(C)cc2[nH]1 4696,Cc1cc(C(=O)NCCC2CCCN2C(C2CCCCS2)=O)ccc1C(F)F 4697,Cc1ccc(C(=O)O)c(-n2cc(CNC(C3(CO)CCCO3)=O)nn2)c1 4698,CN1CCCC(C(N2CCCCC2C(=O)NCC(O)CCO)=O)C1 4699,C(C(Cl)C(C)(F)F)NC1(c2cn(C(C(=O)OC)Cc3ccccc3)nn2)CCC1 4700,N1(C(Cc2scc(CC)n2)=O)CCOC(C(=O)NC(C)CCSC)C1 4701,N1(C(C2CCN(C)C(=O)C2)=O)CCN(C(=O)CC2CS(=O)(=O)C2)CC12CCC2 4702,C(=O)(C(C)(C)C(C)(F)F)N1CCN(C)C(CNC(C2CC23CCC3)=O)C1 4703,Cc1cc(CC(=O)NC2(CCNC(C3CCN(C(N)=O)CC3)=O)CCC2)n(C)n1 4704,N1(C(c2c(-c3cn(CCCN(C)C)nn3)cnn2C)=O)CCc2ncccc2C1 4705,n1(CC(=O)NCCCCCCNC(C2CC2CF)=O)nnc2ccccc2c1=O 4706,C(C1=CCN(C(=O)CC(O)CNC(=O)CC2CCOC2C)CC1)OC 4707,N1(C(CCC=C)=O)CCC(O)CC1C(=O)Nc1csc(C#N)c1 4708,c1(C(=O)NC(CC#C)C(=O)NC2CCCN(C)C2C)ccc2[nH]ccc2n1 4709,C1(CC(=O)NCCC2COCCN2C(c2cc(CO)on2)=O)CN2CCN1CC2 4710,c1(C(=O)NCCCOCCC(=O)NC(CCCCCC)C)cc2cccn2cn1 4711,CCC(C(=O)OC)C(=O)NCCNC(=O)CC1CCC(C)(C)CC1 4712,c1(C(N2C(C)(C)C(O)CC2)=O)nc(=O)c2ccccc2s1 4713,c1(C(N(C)CC2CCCN(C(c3nc(C)oc3)=O)C2)=O)cc(N)c(F)cn1 4714,C1(CNC(CSCC(=O)OC)=O)CCCC(CNC(C2(C)CCC(=O)N2)=O)C1 4715,N1(C(CN(C(c2csc(Cl)c2)=O)CC)=O)CCCC(O)C1C 4716,C1(NC(COc2cccc(C)c2)=O)CCN(C(c2nccs2)=O)C12CCCC2 4717,C1(C(=O)OC)CS(=O)(=O)C2CN(C(=O)NCC3C(C)(C)CCCC3(C)C)CC12 4718,C1(Cn2cc(CC(C)O)nn2)CN(C(=O)Cn2ncnn2)CCO1 4719,CC1CCN(C(=O)CN(CC(F)(F)F)C(=O)C(C2CC2)C2CC2)CC1CO 4720,C(N=c1[nH]c2c(c(=NCC3CCCOC3)[nH]1)CC(C)CC2)c1c(OC)cccc1 4721,c1(CC(C)C)cc(C(N2CC(C)(C(N3CCC(CO)C3)=O)C2)=O)no1 4722,C1(NC(C2C(C)(C(F)F)C2)=O)CC2CCC(C1F)N2C(=O)CC1(C#N)CC1 4723,N1(C(c2cnc(C)c(N)c2)=O)CCCC2CN(C(=O)C3=CCN(C)C3)CC12 4724,C(=O)(CC(C)(C)C(=O)OC)N1CCCC(C(=O)NC2CCN(CCC)C2)CC1 4725,C(=O)(C(C)(C)C(C)C)N1CCC(N(C(=O)CN2C(C)CCC2C)CCC)C1 4726,N1(C(C2C(C(=O)OC)C2)=O)CCC2C(NC(c3cnn(CCF)c3)=O)C12 4727,c1(C(=O)NCCC2N(C(c3nccc(C)n3)=O)CCC2)cnn2cc[nH]c(=O)c12 4728,C(=O)(C(CC)C(C)(C)CC)NC1CCN(C(c2cc(CC)cc(C)c2)=O)C1C1CC1 4729,N1(C(C2OCCN(CC)C2)=O)CCCC2(C1)C(NC(=O)CC(C)(F)F)CCN2C 4730,c1(C(N2C(CN(C(=O)CC(C)COC)CC)CCC2)=O)cc(N)nc(Cl)c1 4731,N1(C(c2ccc(Cl)nc2F)=O)CC2OCCN(S(=O)(=O)c3cccnc3)C2C1 4732,c1(CN2CCC(N3C(=O)CCC3=O)CC2)nc2cc(Br)ccc2o1 4733,c1(SCC(=O)NC2CC(NC(C34CCC(CO3)C4)=O)C(O)C2)cc(F)cc(F)c1 4734,c1(OCC)nccc(C(=O)NCCCCCCNC(=O)Cc2cc(C)no2)c1F 4735,CC(C)CC(CNC(C1(OC(C)C)CCC1)=O)C(=O)N1CCC2CC12 4736,N1(C(CC2CN(C(C)=O)C2)=O)CC(CNC(C2CC(C)(C)CO2)=O)CC(C)(C)C1 4737,C1(C(N2CCC(C(C)NC(=O)Cc3ccc(Cl)nc3)C2)=O)CCC2CC1C2(C)C 4738,C(C)(C(C(=O)NCCC1CCN(C)CC1)C(C)C)NC(Cc1cncc(C)c1)=O 4739,CC1CCN(C(=O)CCC2CCC(=O)NC2)CC1NC(=O)C=CS(C)(=O)=O 4740,C12(CNC(C3C(C)CCC3)=O)CCCC1CN(C(c1ccn(C)n1)=O)C2 4741,N1(C(CCC(C)(C)N(C)C)=O)CC2(CCC2)CC1C(=O)NC1CCOC1(C)C 4742,Cc1ccnc2sc(C(=O)NCC3CCCCC3C(=O)O)c(C)c12 4743,O=C(CN=c1nc(N2CCC(CO)C(F)(F)C2)c2c([nH]1)COC2)NC1CCCC1 4744,C1(NC(=O)COCCCF)COC2(CCN(C(c3coc(Br)c3)=O)C2)C1 4745,c1(NC(c2nc(C)cs2)CC)nc(C)cc(=NCc2cccc(O)n2)[nH]1 4746,c1(C(=O)NCCn2cc(C(N(CCC(=O)NC)CC)=O)nc2)cccc(C)c1O 4747,Cc1cc(C)nc(N(C2(C#N)CCNC2)C(C2CCC(=O)NC2)=O)n1 4748,N(C1CCOc2c(F)cc(F)cc21)C(C(C)Oc1ccccc1CC(=O)O)=O 4749,c1(C(=O)NCC2CCC2NC(C2CCCS2)=O)cscc1F 4750,N1(CCCCOC)CCCCC(NC(c2cnnn2-c2ccccc2)=O)C1 4751,C1(NC(c2c(C)n[nH]c2C)=O)CC2CC(NC(C3CCS(=O)(=O)N3)=O)CC12 4752,S(=O)(=O)(c1cccc(Cl)n1)SCCC(N1CC(c2ccccc2)(O)C1)=O 4753,C1(C(=O)NCCC2CN(C(C3(S(N)(=O)=O)CC3)=O)C2)CC2CCC1C21CC1 4754,n1(CC)ncc(C(=O)NC2(CNC(=O)C(C)C#N)CCOC2)c1C 4755,CC(C(=O)NC1CCCC1)NC=O.C1(c2nc[nH]n2)(NC(C=CC)=O)CCC1 4756,Cc1cc(C(N2CCOC(C(N(CCCc3ccccc3)C)=O)C2)=O)nn1C 4757,C(=O)(C1=C(C2CCOCC2)N(C)C(=S)NC1c1cccc([N+](=O)[O-])c1C)OCC 4758,C1(C)(CC)CC(NC(=O)Cc2cc(C)[nH]n2)CN1C(C1(NC(N)=O)CC1)=O 4759,n1(CC=C)c(N(CC(C)CC)C)nnc1C1COc2ccccc21 4760,CC1CC(C(=O)N2CC(O)(C(C)(C)CNC(C3CCCC34CC4)=O)C2)=NO1 4761,C1(NC(c2c(SCC)cccc2)=O)C2CC1N(C(c1cnc(S)[nH]1)=O)C2C 4762,C(CN=c1cc(F)nc[nH]1)(c1ccccc1F)NC(C(C(C)C)C)=O 4763,N1(C(c2ccsc2Br)C(=O)NC2CCC2)CCC2(C1)OCCO2 4764,C1(CCC)CN(C(=O)C(=O)NC2CC(C(=O)NC)C2)C1 4765,c1(C(N2C3CN(C(C(C(CC)C)O)=O)CC2C3)=O)onc2ccccc12 4766,C12(NC(C(C)Cn3ccnc3)=O)CCC(F)(F)CC1CN(C(=O)C(C)(C)CF)C2 4767,C1(CC)CCC(C(=O)N(C2CCC(NC(c3cccc(N(C)C)n3)=O)C2)C)CC1 4768,c1(NC)ccc(C(N2CC3CCCC23)=O)cc1[N+](=O)[O-] 4769,C(=O)(C1CCc2cc(F)ccc21)NC1(C)CCN(c2cc(C(C)C)nc(Cl)n2)C1 4770,c1(CC(N2CC(NC(c3n[nH]cc3Br)=O)C3C2C3)=O)cccc(F)c1O 4771,c1(C(N(c2ncncc2Br)C(C2CCCNC2)C)=O)ccc2c(c1)C(=O)NCC2 4772,C1(CC(=O)NC(C#C)C(C)C)N(C(=O)CC2CCC(C)CO2)CCC1(C)C 4773,N1(C(C2C=C(C)CS2)=O)CC(O)CC1CNC(C1CC2(CCC2)C1)=O 4774,CC(C)(C)CCCC(=O)NC1CCC(NC(=O)CCc2c[nH]c3ccccc23)C1 4775,C1(C(N2CCC(OCC)C2)=O)CC2(CC2)CN1C(=O)C(=O)C(C)CC 4776,CC1(CNC(=O)CN(C(=O)Cc2ccsc2)C2CC2)CCCC1 4777,N1(C(c2n[nH]c(C)c2C)=O)CC(NC(=O)C(CC2CC2)CC2CC2)CCC1C 4778,Cc1cc(C(N2CCC(N(CCO)C(C3(C)CCC(=O)NC3)=O)C2)=O)ccc1F 4779,N1(C(C(SC)SC)=O)CCCCC(N(C)C(c2ccc(F)c(F)c2)=O)C1 4780,c1(OC)cc(C(=O)NCCNC(c2c(C3CC3)cnn2C)=O)cc2cn(C)nc12 4781,C(CC(C)CCNC(=O)C=C1CCC1)NC(c1cn(CCOCC)nn1)=O 4782,N1(C(C2C(C)(C)C2CNC(=O)Cc2ccco2)=O)CCC2(CC1)CSC2 4783,C1(CNC(=O)NCCC2CCCS2)CCCN(c2ccccn2)C1 4784,c1(OC)ccc(CNCCCCC2CC2C)cc1C#N 4785,C=C(C)C1OCCC1C(=O)NC(CC)CC(=O)NC1CCN(C)C1(C)C 4786,C1(NC(c2nccc(OC)c2OC)=O)C2CCC1CN(C(c1snnc1C)=O)C2 4787,c1(OC)cccc2[nH]cc(CC(=O)N(C)CC3(O)CCC(F)(F)CC3)c12 4788,C(=O)(C(F)(F)C(F)(F)F)N1CCC(N(C)C(=O)Nc2cc(C(F)(F)F)ccc2O)C1 4789,C=CCC(C)(C)CNC(C1CCN(C(=O)CP(C)(C)=O)C1)=O 4790,CC1C(NC(=O)Cc2cnsc2)CC2CCC1N2C(=O)C(F)(F)c1cnccn1 4791,N1(C(c2c(C)n[nH]c2)=O)CCN(C(=O)C=CC=CCO)CC1c1ccnn1C 4792,N1(C(CC(CN(C)C)(C)C)=O)CC2CCCCC2(NC(C2OCCC2(C)C)=O)C1 4793,c1(C(N2CCC23CCCC3)C(=O)NCCOC)cc(OC)cc(C(F)(F)F)c1 4794,c1(OCC)c[nH]ccc1=NC(=O)CSC1CCCCN1 4795,C(c1cc(Cl)ccc1Cl)=CC(N1CCN(C(C2CCC(O)C2)=O)CC(CO)C1)=O 4796,C1(C(=O)NC(C2CCN(c3nc(C)nc(O)c3C)C2)C)CCC2(CC1)CC2(F)F 4797,c1(CNC(C(CO)NC(C2C(C)CC2)=O)=O)ccc2c(c1)CC2 4798,C(C(C(=O)NC1CCOCC1)N(C1CCC1)CC1CC1)(C1CCC1)OC 4799,CCC(C)CC(=O)C(=O)NC(C1CC1C(=O)NCc1ccc(C2CC2)o1)C 4800,C1(CNC(C(C(C)C)OCC)=O)CC12CCN(C(=O)C(F)(F)c1cncs1)CC2 4801,c1(N(C(C)=O)C)ccccc1C(=O)N(CC(C)CNC(C1CC(N=[N+]=[N-])C1)=O)C 4802,CCCCC(C)CCC(=O)NC1COCC1NC(c1cc(Br)cs1)=O 4803,CC1CN(C(=O)OC(C)(C)C)CCC1N(C)CC1(O)CCOCC1 4804,C(c1ccc(Cl)c([N+](=O)[O-])c1)=CC(=O)NC1CC2(CNC2)C1 4805,C(CCCCC(=O)N1CCN(C(c2cnc(C)nc2)=O)C(C2CC2)C1)NC(C)=O 4806,c1(C(=O)NCC2N(C(C(C)OCc3ccccc3)=O)CC=C2)c(O)cccc1F 4807,C(c1cncn1C)=CC(=O)N(CCC(=O)N(CC(O)C1CCC1)C)CC 4808,N1(C(C(COC)NC(C)=O)=O)CCC2CC1CN2C(c1cccc(C)n1)=O 4809,c1(SC)ccc(C=CC(=O)NCC2CC(NC(=O)CCNC(C)=O)C23CCC3)s1 4810,C1(C(=O)NCC2(C)COCCO2)CCC2(CCNC2)CC1 4811,CC(C)C(CC(=O)NCC(F)CNC(c1cocn1)=O)c1ccccc1 4812,CCC(CC)CC(F)C(=O)NCC=C1CCN(C(c2ccc(C(C)C)s2)=O)CC1 4813,Cc1cccc(NC(=O)NCC(c2ccc(C3CC3)cc2)(C)C)c1F 4814,C1(CNC(COCC)=O)CN(C(C2(CC(C)=O)CC2)=O)CCC1(C)C 4815,C1(CC(=O)N(CCC)C2CC2)CN(C(C2CC(C)=NO2)=O)CC12CC2 4816,c1(CNC(CC2(CC)CCC2)=O)cc(C(=O)N(C2CC2(C)C)C)on1 4817,CCCCC(C(=O)NCc1ocnc1CC)NC(c1cc(C)c(C)[nH]1)=O 4818,c1(CCNC(C=CC(C)(C)NC(c2cc(O)cs2)=O)=O)ccncc1F 4819,C1(CCOC)CCC(C)N(C(c2sc(Cl)cc2Cl)C(=O)Nc2cccc(F)c2)C1 4820,CCC(C)CC(CO)NC(=O)CC(CC)N(C)C(C1CC(=O)N(C)C1)=O 4821,Cc1nc2ccc(NC(C3CC(F)CN3c3ncnc4sc(Br)cc34)=O)cc2o1 4822,C(=O)(C(F)CCC(C)C)NCC1N(C(CC2CCC(OC)CC2)=O)CC1 4823,Cc1n[nH]c(=NC2CCCC(NC(c3cnn(C4CCCC4)c3C)=O)C2)s1 4824,c1(C(=O)NCCC2N(C(C=C(CCN(C)C)Cl)=O)CCC2)c[nH]cc(C)c1=O 4825,N1(S(CC)(=O)=O)CCCCC1C(N1CC=CC(NC(=O)C#CC2CC2)C1)=O 4826,C1(NC(CCCC(C)C)=O)CCN(C(c2cc(O)cc(=O)o2)=O)C12CCCC2 4827,C1(CNC(C2(CCC)CC2)=O)CC2(CCN(C(C3(C)C=CCC3)=O)CC2)C1 4828,c1(C(N2CCOC(C3CCOCC3)C2)=O)[nH]cc2c1CCC2 4829,c1(C(=O)NCC2C3CN(C(CCCCCC)=O)CC32)cc2n(n1)C(C)CCC2 4830,c1(OC)c(C(=O)NC(CN(C)C)C(=O)NCC2CC(F)C2)cnn1C 4831,c1(C(=O)NC(C)CC)cc(N(CC=C)CC)c(OC)cc1-c1ccc(CC)cc1 4832,N1(C(C(C)SC)=O)CCC(F)(F)C(CNC(C2(C)CC(C)(C)C2)=O)C1 4833,C1(NC(C2CC3CCC2C3)=O)CC2CCC1N(C(=O)CN1CCCS1(=O)=O)C2 4834,C1(CNC(C(CC)N(C)C)=O)CC2COCC2N1C(c1cc2cccnc2s1)=O 4835,C12(CNC(c3ccc(O)nc3)=O)CCC(CN(C(=O)C=Cc3cscn3)C1)C2 4836,N1(C(C(CCCC)O)=O)CC(NC(c2ccncc2)=O)C2CCCC2C1 4837,c1(C(N2C3CN(C(c4c(CC)scc4)=O)C(CC3)C2)=O)ccnc2c1CC(=O)N2 4838,c1(C(N2CCOCC(NC(CC3(CSC)CC3)=O)C2)=O)cc(O)cc(C#N)c1 4839,C=CCC(C(=O)NC(C)CCNC(C1(C2CCCO2)CCCC1)=O)C(C)C 4840,C(CC(C)C(=O)NCC1CCN1C(=O)CN1CCCCC1)OC 4841,C1(CCNC(C2CC(c3cn(CC(F)(F)F)nn3)C2)=O)OCCCO1 4842,CC1CN(C(c2c(F)cccc2Cl)=O)CCN1C(c1ccc(C2CC2)cc1)=O 4843,N1(C(C2CC(=O)N2)=O)CCOCC12COCCN(C(C1C3CCCCCCC13)=O)C2 4844,N1(C(C=Cc2ccc(C)nc2)=O)CC2(CCN(C(=O)CC3CCOC3C)C2)C1 4845,C(CCCCC(=O)N(C1CCC(C(=O)NCC(C)C(=O)OC)C1)C)SC 4846,c1(C(=O)NCC(C)=CC(=O)NCCN(CC(C)(C)C)C)cnc(C)c(C)c1 4847,CC(C(F)(F)C(F)(F)F)NC(=O)Nc1ccc(Br)c(Cl)c1F 4848,S(=O)(=O)(c1ccc(SCc2ccc(CC(=O)O)cc2)cc1)NCN(C(C)C)C 4849,c1(NC)ncc(C(=O)N(C2CCCCC2)CCNC(C2(CO)COC2)=O)cc1Cl 4850,CC(C)CCCCCC(=O)NCC12CCCCC1N(C(=O)C1=COCCO1)CC2 4851,n1(CC(=O)NC(c2cnn(C)c2)C(=O)NCCC2C(C)C2)[nH]cnc1=N 4852,C(=O)(CCCC(N)=O)N(C(C)CCNC(=O)CC1CN(C)C1)C 4853,CCCCCC(O)C(=O)N(CC(N1CC(c2cc[nH]n2)C1)=O)CC1CC1 4854,c1(OC)cc(C(=O)NCC(CO)NC(C2(c3ccc(C)nc3)CC2)=O)ncn1 4855,c1(NCc2nc(C)[nH]n2)nc(N2CCC(NC(C)=O)C2)c2ncn(C(C)C)c2n1 4856,C(=O)(C(O)C(F)(F)F)NCC(C)(C)NC(c1cn(C)c(O)n1)=O 4857,c1(N2CCC(C=C)CC2)nc2c(c(=NCC3CCC=CCCC3)[nH]1)CCC2 4858,c1(C(c2ccccc2)Nc2c(C)nc(C)[nH]2)c(C#N)c(C2CC2)nn1C 4859,C1(C(CC)NC(CCC=C)c2nnnn2CC2CC2)CCC(F)(F)CC1 4860,c1(CC(N2CCC(F)(COC)C2)=O)cccc2ccccc12 4861,C(=O)(CC1OCc2ccccc21)NCC(C)NC(c1n(CC)nnc1)=O 4862,C1(C(=O)OC)CC2CC(NC(=O)Cc3cnc(C)nc3O)C2C1 4863,C(CC(=O)NC1CCC(CNC(=O)C(C)CC2CCC2)C1)(OCC)OCC 4864,N1(C(C2C(C)(C)CO2)=O)CC2CC(NC(=O)CCCC3CCCCC3)CC2C1 4865,c1(C(=O)NCCN(C(c2[nH]nnc2C(F)F)=O)CC)cnc(O)n1CC 4866,N1(C(CCOCCCOC)=O)CCC(C(F)F)(CNC(c2sccc2Cl)=O)C1 4867,Cc1noc(N)c1C(N1CCC(NC(c2csc(C(F)(F)F)c2)=O)C1)=O 4868,c1(C(=O)NCCN(C(=O)Cc2ccc(Oc3ccccc3)cn2)C)nnc(S)n1C 4869,N1(C(CC(CC)C2CC2)=O)CC(NC(C2CCN(OC)CC2)=O)C2(CC2)C1 4870,CC1CC(c2cn(-c3ccncc3)nn2)CCN1CC(N1CCC(O)CC1)=O 4871,C1(C(N2CCC(NC(Cc3cccc(C#N)c3)=O)CC2)=O)CCc2ncnn2C1 4872,S(=O)(=O)(c1cccc(Br)c1)C(=O)NC(C)C(=O)NCc1ccc2ccccc2c1 4873,C12(OC)CN(C(=O)Cc3ccnc(C(=O)OC(C)(C)C)c3)CC(C(=O)O)(C1)C2 4874,N1(C(C(CC)(C)OC)=O)CCCC(CC)(NC(=O)CCc2ccccc2F)C1 4875,CC(C)S(=O)c1ccc(C(=O)NC2CN(C(c3c[nH]c(=N)o3)=O)CC2O)cc1 4876,N1(C(c2sc(C)c(Br)c2C)=O)CCC(C2CC2)C1CNC(=O)CC1CC1 4877,n1(CCC(=O)NCC2COCCN2C(C2CCC2)=O)cc([N+](=O)[O-])cn1 4878,c1(C(=O)OC)ccc(S(=O)(=O)NC2CCCN(C(c3cncs3)=O)C2)cc1 4879,C1(CC=C)(NC(=O)CC(O)CCSC)CCCN(C(c2ccc(C=CC)o2)=O)C1 4880,N1(C(C(CC=CC)CC)=O)CC2OCC(NC(=O)CCCCCCC)C2C1 4881,c1(C(N2CCC(C(N(CCOC)C(C)C)=O)CC2)=O)nccc2ccccc12 4882,CC1CN(C(=O)C(CC(N)=O)NC(c2ccc(F)s2)=O)C(C)CO1 4883,c1(NC(C2(CC=C)CCCN2C(=O)C=C2CCC2)=O)cccc2cccnc12 4884,c1(CO)ccnc(N(C2CCSC2)CC2CCCO2)c1I 4885,c1(-c2n(CC(C)(C)C)nc(CCOc3ccccc3)n2)cc2c(nn1)CCOC2 4886,C(CC)(CCCC(=O)NCC(C)(C)CCOC)NC(c1cnc(CC)o1)=O 4887,c1(C(N2CCCN(S(=O)(=O)c3cccs3)CC2)=O)noc2c1CCCC2 4888,C(CC(C(=O)NCCc1ccncc1)NC(=O)C1=NOCC1)OCC 4889,Cn1cc(C(=O)NC2CCCN(C(=O)CCC3CCCCC3)C2)c(O)nc1=O 4890,c1(OCC(=O)NC2(CNC(CSC)C)CCOC2)cc(C)ccc1Cl 4891,CC1CCC(C)(C(N2CCCCC2CNC(=O)Cc2cccnc2F)=O)CC1 4892,c1(NC(C(C)C)=O)ccc(C(=O)NC2CCN(C(=O)C(C)(O)C3CC3)C2)cc1 4893,c1(C(C)=O)ccccc1C(=O)NCC(C)NC(=O)CCCCN(C)C 4894,C1(C(=O)NCC=C2CCN(C(C(CC)(C)O)=O)CC2)CC(C(C)C)=NO1 4895,c1(OCc2nc(-c3nn(CC)c(C)c3)n(C3CC3)n2)ccc(C)c(Br)c1 4896,Cc1c(Cl)cc(C(=O)NCC(C)NC(=O)CNC2CCOC2=O)cc1Br 4897,CCS(=O)(=O)c1ccc(C(N2CCC(C(F)F)C2)=O)cc1 4898,C12(C(=O)NC(c3ccnn3C)C)CC1CCN2C(=O)Cn1cnnn1 4899,N1(C(c2ccc(CC(C)(C)C)cc2)=O)CCC12CN(C(C1SCCCS1)=O)C2 4900,c1(NC2(CNC(C3N(C(C)C)C(=O)CC3)=O)CCCC2)ncc2ccccc2n1 4901,c12ccc(cc1)CNC2.CCCC(C)(c1nnnn1C)SC1CCCCO1 4902,CCCCC(CC(=O)N(C(C)CC(C)CC)C)NC(=O)CC1(C)CC1 4903,N1(C(C2(C)CC(OC)(OC)C2)=O)CC2(CCC(CNC(=O)C(O)C(C)C)O2)C1 4904,c1(OC)cc(C(=O)Nc2c(Cl)ccnc2Cl)cnc1-c1ccnc(F)c1F 4905,C1(NC(C=CC(C)C)=O)CCCCN(C(=O)CC2CCCC(C)(C)O2)C1 4906,c1(OCC)ccc(C)nc1C(=O)NCC(F)CNC(C1CC1C(F)(F)F)=O 4907,c1(CC(N2CCCC(NC(CCCNC(N)=O)=O)C2)=O)cc(Br)ccc1F 4908,c1(OCC(N2CC(F)(CNC(c3c(C)con3)=O)C2)=O)c(C)cccc1Cl 4909,C1(CC(=O)N(CCCNC(=O)CCn2ccnc2)CCO)CCCCCC1 4910,C1(F)(CNC(c2cc(C)nnc2)=O)CCCN(C(=O)CC2(O)CCCCC2)CC1 4911,N1(C(=O)NC)CCC(C(N2CCCC(CNC(=O)CSC(C)C)C2)=O)CC1 4912,CN1CCN(C)C(C(=O)NC2CCC2NC(=O)CC#N)C1 4913,c1(C(=O)NC(C(C)NC(C2CCS(=O)(=O)C2)=O)CO)ccnn(C)c1=O 4914,CC1(C(N2CCCC(NC(c3coc(CC4CC4)n3)=O)C2)=O)CC2(CCC2)C1 4915,N1(C(C2(C)ON=C(C)C2)=O)CCN(C(c2cnc(O)n2C)=O)C(CC2CC2)C1 4916,N1(C(C(C=C=C)C)=O)CC2CCN(C(c3cc(C)oc3C)=O)CC2C1.[SH](C)(=O)=O 4917,c1(C(=O)NC2C3CN(C(C4(n5cccn5)CC4)=O)CC23)c[nH]c2cccnc12 4918,N1(C(c2cnc(C)o2)=O)CC2CCC(NC(c3cccc(F)c3Cl)=O)CC2C1 4919,C=CCCCC(C(=O)NCc1ccc(C)nc1O)NC(=O)CC(O)CC(C)C 4920,c1(NC(C2CC(F)CCN2C(C2C3CCC(C3)C2)=O)=O)ccc(CO)cc1O 4921,C(=O)(C(O)CC[S+](C)C)N1CCC(NC(c2c(C)oc(C(C)(C)C)c2)=O)C(O)C1 4922,C#CCC(C(=O)N1CCC(N(C(=O)CN2CCC(C)(O)C2)CC#C)CC1)C1CC1 4923,C1(CNC(C(c2ccoc2)NC(C2CSCC(=O)N2)=O)=O)CC(O)C12CCC2 4924,C1(C(=O)NCC=CCNC(C(N2CCC(O)CC2)C)=O)CCCC(CF)C1 4925,Cc1cc(C(=O)NC2(c3ccccc3)CN(C(=O)C=C3CCOCC3)C2)n[nH]1 4926,C1(C(=O)NCC2(C(=O)NC(c3ccncc3)C)CC(C)(C)C2)CCC(C#N)CC1 4927,C1(C(N2C(CN(C(=O)CC3CCC34CCC4)C)CCC2)=O)CCC2(CC1)CC2 4928,N1(C(CS(=O)(=O)NC)=O)CCCC(N(C(=O)CCc2cnc(C)s2)CC)CC1 4929,C(=O)(CCCCCN=[N+]=[N-])NCCC1(OC)CN(C(=O)COCC2CCC2)C1 4930,Cc1nn(C)c(C)c1CC(C)C(=O)NCC(CO)NC(=O)CN1CCCCCC1 4931,c1(CC)conc1C(=O)NCC=CCNC(C1(O)CC(c2ccccc2)C1)=O 4932,n1(CC)cc(C(=O)NC(C)C(C)NC(c2cc(C(F)(F)F)ns2)=O)nn1 4933,c1(C(N(CCN(C(c2c(CC)oc(C)c2)=O)CC)CC)=O)cc2n(c1)CCC2 4934,c1(C(=O)NC2CC(NC(c3cc(CC)c(CC)o3)=O)C2)c(F)cc(Cl)cc1Cl 4935,N1(C(C2CN(C(C3(COC)CCC3)=O)CC23CCC3)=O)CCCC(N=[N+]=[N-])CC1 4936,CCCCC(O)C(=O)NCCN(C(c1ccc(OC)cc1F)=O)C(C)C 4937,N1(C(CCc2n(C)ncc2)=O)CCOC(CCNC(C2CC2(C)C(F)F)=O)C1 4938,c1(CC)ccc(NC(=O)C(c2cccnc2F)(C)C)cc1Cl 4939,Cc1cc(C)c(C(=O)NC(C)C(C)NC(c2coc(N(C)C)n2)=O)cc1N 4940,CC(O)CC(=O)N1CC(N(C)C(C2CSC2)=O)C1 4941,C12(NC(CC3(C)CC3)=O)CC3CC(C1)CC(NC(C1CCCC(O)C1)=O)(C3)C2 4942,Cc1cc(O)cc(C)c1CC(=O)NCC1(CNC(=O)Cc2ccccn2)CCC1 4943,c1(C(=O)NCC=C)cccc(S(=O)(=O)NC(C)CNc2cccnc2)c1 4944,CC1CCCCC1(CNC(=O)CCn1cnccc1=O)NC(C1CC(=O)N1)=O 4945,c1(NCC(=O)N(CCCNC(=O)CNC(C2CCCSC2)=O)C)cccnc1 4946,N1(C(CC2(C(=O)OC)CC2)=O)CC(=O)NCC1C(C)C.C(CCN)O 4947,N1(C(C(CC=C)C)=O)CCCCC(NC(c2ccc(N3CC=CC3)cc2)=O)CC1 4948,C1(NC(C2N(C)CCC2)=O)CN(C(=O)CCc2ccc(=N)[nH]c2)CC12CCC2 4949,N1(C(c2ccc(C#C)cc2C)=O)CCC2CCN(C(c3cocn3)=O)C2C1 4950,c1(C(=O)NCC(CC)(C)NC(=O)C(C)NC(=O)COC)cc2cncn2c(O)n1 4951,CCCCS(=O)(=O)NC(C)C(N1CC(N(C)C(c2nn(C)cc2Cl)=O)C(O)C1)=O 4952,N1(C(CNC(CCCCC)=O)=O)CCN(C(=O)C(C)CO)CC1C(F)F 4953,C(=O)(CC(C)(C)C(F)F)N1CC(C2CN(C(CN(C(C(C)C)=O)C)=O)C2)OCC1 4954,c1(C(N(C(CNC(C2(Cl)CC2(F)F)=O)C2CC2)C)=O)cnc2c(Cl)cccn12 4955,C1(C(=O)NCc2nc(C)sc2)C=CCN(C(=O)C(F)CC2CCOC2)C1 4956,N1(Cc2cn(C(C)C(=O)NC3CC(CN4CCCC4C)C3)nn2)CCCOCC1 4957,N1(C(C2(CCC=C)CN(C(=O)CC=CC)C2)=O)CC2CCC1C(O)C2O 4958,c1(C(N2CCC(CCNC(c3c(C)ccs3)=O)C2)=O)nc2c(s1)COCC2 4959,C(=O)(C1CCC(NC(=O)Nc2cc(Cl)cc(Cl)c2)c2ccccc21)OC 4960,Cc1ccc(O)cc1C(N1CC2CC(C1)N2C(c1ncoc1C(C)C)=O)=O 4961,N1(C(=O)CC2CC3(CCO2)CC3)CCC2C(C1)CN2C(=O)Cc1cnoc1 4962,N1(C(CCN(C(=O)COC2CCOC2)CCCO)=O)CCCC2(CCCO2)C1 4963,CCCCC(C)C(=O)NCC12COC(CNC(=O)CC3COC(C)(C)CO3)(C1)C2 4964,C1(CC)(NC(=O)C=CSCc2ccco2)CN(C(=O)CNC(c2ccoc2)=O)C1 4965,c1(CNC(=O)NCC(c2cccc(O)c2)(C)C)ccc(Br)c2nsnc12 4966,c1(C(N2C3(C(=O)NC4C(OC)C(O)C4)CC3CC2)=O)cccc(F)c1F 4967,c1(CNC(C2(CSC)CC2C)=O)cc(O)nc(CNC(=O)COC2CCCC2)n1 4968,c1(OC(C)C)ccc(C(=O)NCCCN(CCO)C(c2cn(C)nc2Cl)=O)cc1 4969,N1(C(C=CC)=O)CCCC(O)(CNC(=O)C(F)(F)CC2CCCO2)C1 4970,c1(C(=O)NCCSCC)n[nH]c2c1CN(C(c1ncc(C)cc1F)=O)C2 4971,CC1CC2(CCN(C(=O)C(C)n3cncn3)CC2)CN1C(=O)Cc1ccncc1 4972,c1(C(=O)NC2CCC(NC(c3c(Cl)nc(N(C)C)s3)=O)CC2)ccc(=O)n(C)n1 4973,C1(=O)C2=C(C)N(C(=S)NC2c2cc(I)ccc2Br)C12CC2.C(=O)OC 4974,C1(C(=O)NCCC(CCC)C2CC2)CC2(CCC2)CN1C(=O)C1=NOCC1 4975,C(C)(CCN=c1c(Cl)c[nH]cc1[N+](=O)[O-])NC(CCCc1cc(C)no1)=O 4976,c1(NC)ncccc1C(=O)NCC(C)(C)NC(c1ncc(OC)cn1)=O 4977,c1(C(=O)NC2(C)CCN(C(C(C=C)(C)O)=O)C2)cc(C)nc2c1cnn2CC 4978,C(=O)(C1CCCn2ccnc21)NC1C(C)C2CCC(C1)N2C(C1CC1(C)Br)=O 4979,N1(C(c2nc(COCC)sc2)=O)CCOCC1CN(C(=O)CC1CCOC1)C 4980,C(C)(CCC(C)C)N(C(C1C(C)=CCS1)=O)C 4981,N1(C(CC(C)CNC(C2(C)CC(C#N)C2)=O)=O)CC2CN(C)CC2C1 4982,c1(CNC(C2OCCN(C(CCCN(C)C)=O)C2)=O)ccc(F)c(O)c1 4983,c1(NC(C)CCC(F)(F)F)[nH]c(=NC2CSc3ccccc32)nc2sccc12 4984,CC(CNC(=O)Nc1ccccc1OCCNC)CC(F)F.C1(O)CCCC1 4985,C1(C2CCN(C(=O)C=Cc3ccc([N+](=O)[O-])s3)C2)(NC(CCSC)=O)CC1 4986,CC(=O)CCCC(=O)N1CC(NC(C2CCCN2C(=O)OCc2cccs2)=O)C1 4987,C1(NC(=O)NC2CCC3(C(=O)OC)C2C3)CCC2OCCC2C1 4988,C12(NC(c3ccncc3Cl)=O)CCCCC1N(C(c1cncc(Cl)c1)=O)CC2 4989,CN1CCOC2CN(C(C3(CNC(=O)C(=O)NCC4CC4)CC=CC3)=O)CC12 4990,C1(C(=O)NCCCNC(=O)CC2CCC3(CCC3)OC2)CC2C=CCC(C1)C2 4991,c1(C(=O)NCC2CN(C(CCC(C)C)=O)CC2O)cn2c(n1)C(C)CCC2 4992,C1(C)(NC(c2cc(NC(CC3(OC)CCC3)=O)no2)=O)CCCC1C 4993,C1(C2CCC2)(NC(C2C=CCCN2C(=O)CCCc2cnn[nH]2)=O)CC1 4994,Cc1cc(C(=O)NC2CN(C(c3ccc(Br)cc3)=O)C2)nnc1C 4995,C1(CC=C)(NC(=O)C(F)=CC)CCCN(C(=O)Cc2cc(Br)cs2)C1 4996,Cc1cncc(C(N2CCCCC2CCCNC(=O)CSc2ccncc2)=O)n1 4997,c1(C(N(C)CC2CCN(C(=O)CC3CC(=O)NC3=O)C2)=O)ccnc2c1CCO2 4998,C1(C(N2CCC(CCC)C2)=O)COCCN(Cc2cccc(OC)c2Cl)C1 4999,c1(OC)cc(C)ccc1CNc1cnc(F)cc1C(=O)N(C)CCO 5000,C1(O)(C(C)NC(=O)C=CC2CC2)CCN(C(c2cc(CC3CC3)no2)=O)C1 5001,C1(CNC(C(CC)n2cncn2)=O)CCN(C(c2c(C)noc2C)=O)C12CCC2 5002,Cc1cnoc1C(=O)NCC1(CN(C(=O)Cn2cnc(C(N)=O)n2)C)CC1 5003,C(=O)(CC(C)(C)n1cc(-c2ccc(Cl)cn2)nn1)NC(C)COC1CCCC1 5004,C12(NC(c3cc(C)[nH]n3)=O)COC(CNC(=O)C(N3CCNC3=O)C)(C1)C2 5005,N(S(=O)(=O)N1CCC(C)C1)CCC1(NC(=O)OC)CCC1 5006,C1(CNC(C2(N(C(c3ccc(COC)o3)=O)C)CC2)=O)CC(O)C(O)C1 5007,C(=O)(CC(C(F)(F)F)c1ccon1)N(C1CCN(C(CN(C)CCO)=O)C1)CCO 5008,c1(C(=O)NCC(C(=O)NCCSCCO)N(C)C)cccc(F)c1N 5009,C(=O)(CC(O)c1cnc(Cl)s1)N(CCNC(C1(CCC=C)CC1)=O)C 5010,C(C(C(=O)NOCC(=O)OC)NC(=O)C(O)CCN(C)C)OCC 5011,CC1(CNC(=O)NCCC2CCCCO2)Cc2ccccc2C1 5012,C1(NC(N(CC(C2CCCC2)O)C)=O)CCC2(CCCNC2)C1 5013,c1(OC)ccc2[nH]nc(CNS(=O)(=O)Cc3cccc(Cl)c3OC)c2c1 5014,c1(C(=O)OCC(=O)N(C2CCS(=O)(=O)C2)CC#C)cccc(C(C)(C)C#N)c1 5015,C1(CNC(c2cccc(C3(C)CC3)c2)=O)CC2(C1)CN(C(=O)C#CC1CCC1)C2 5016,N1(C(Cn2nnc(C)n2)=O)CCn2c(CNC(C3COCC(C)O3)=O)nnc2C1 5017,C1(NC(CCCc2onc(CC)n2)=O)CCC(C)(CNC(=O)Cc2ccco2)C1 5018,c1(-c2ccc(C3(C(=O)Nc4nc(Cl)ccc4O)CC3)cc2)cc(Cl)c(Cl)cc1Cl 5019,N1(C(C(C)CC2CC2)=O)CCC(CNC(=O)CC2CCCOC2)C(C2CC2)C1 5020,C(=O)(C(C)C(F)F)NCC(N(C(Cc1cc(C)no1)=O)C)C1CC1 5021,C(=O)(C(F)C(C)CC(C)(C)C)N1C(C2(NC(COC(CC)C)=O)CC2)CCC1 5022,c1(C(N2CC(CNC(CC(=O)OC)=O)C3(C2)CC3)=O)ccccc1N=S(C)(C)=O 5023,c1(C(C)C)ccccc1C(=O)NC(C)(C)CN(C(=O)CC1CCN(C)C1)C 5024,c1(C(=O)NC(C)C(C)NC(=O)COc2ccsc2Cl)ncoc1-c1ccon1 5025,c1(C(=O)NC(CC=CC)C(=O)N2CCC(C)CC2)ccc(C)cc1C 5026,C1(COC)(CNC(=O)C(C)(C)n2cccn2)CN(C(c2n[nH]cc2C(C)C)=O)C1 5027,c1(C(C(=O)NC2CCN(C(C(C)N3CCC3)=O)C2)=O)ccc(O)cc1 5028,N1(C(CC2CCC(=O)NC2=O)=O)CCC(C2(NC(=O)CN3CCSCC3)CC2)C1 5029,C(=O)(C1CCc2c[nH]nc21)N1C(CNC(c2cccc3nccn23)=O)C=CC1 5030,C1(N(C(=O)C(=O)Nc2ncsc2Br)CCOC)CCCCCC1(C)C 5031,c1(C(N2CC(CC(C)NC(C(CC)C(C)C)=O)C2)=O)cc([N+](=O)[O-])cnc1N 5032,C12(OC)CCC(C(=O)NC3CCCCC3NC(=O)CC34CCCC3C4)(CC1)CC2 5033,C1(NC(C(C)OCCCC)=O)CN(C(=O)C(c2ccccc2)C)CC(C)(C)C1 5034,CC(C)CC(C)(O)CNC(=O)CNC(=O)Cc1ccc(C#N)cc1 5035,N1(c2ncc(C(C)(C)O)cn2)CCCC(C)(C)C1CNC(=O)CC1CC2(CC2)C1 5036,CCCCCCC(=O)NC1CC2(C1)CN(C(=O)C(C)C(C)c1ccc(F)cc1)C2 5037,c1(N(CC)CC)ccc(C(=O)NC2CC(NC(c3ccoc3Br)=O)C2)cc1 5038,C(=O)(C1c2ccccc2CN1Cc1snc(Cl)c1Cl)N1CC(c2n(C)cnn2)C1 5039,C1(CNC(c2c(OC)csc2)=O)CCCCN(c2cc(C)nc(CO)n2)C1 5040,c1(C(=O)NCC(CCOC)NC(C(CC)OC)=O)cccc(Cl)c1C(F)F 5041,C(N=c1[nH]c(C)cc(=NCC(C)N2CCC(C)CC2)[nH]1)C1CC(OC)C1 5042,c1(C(=O)NC2(CNC(c3cnn(C)c3C3CC3)=O)CC2)cc(C(F)F)cc(Cl)c1 5043,C(=O)(CC(C)COC)N1C(CC(N2C(CCC=CC)CCC2)=O)(CC)C1 5044,CCC(C(=O)NC(C)CN(C(=O)Cn1ccc(Br)n1)C)N(C)C 5045,c1(CNC(C2CC(F)CN(c3ncc(C(F)F)cn3)C2)=O)cccc(F)c1O 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5064,C(=O)(C1=C(F)CN(C(=O)CC2(O)CCC2)CC1)NCC1(SC)CCC1 5065,N1(C(COCc2cccc(C)c2)=O)CCCC12CCN(C(c1ncoc1C)=O)C2 5066,C1(NC(=O)C(c2ccccc2)F)CCN(C(=O)CC(O)c2cnc(Cl)s2)CC1 5067,O=C1NC2(NC(N3CCC(Cc4ccccc4)C34CCC4)=O)CC3CC1C2C3 5068,C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CC(NC(COCC)=O)C(F)CC1 5069,CCC(C)C(C(=O)NC(C)(C)C=CC(=O)NC1CCCC1)OC 5070,Cc1n[nH]c(C)c1C(=O)NCC1CN(C(=O)C(C)Oc2ccccc2F)CCO1 5071,C1(C#CC(=O)N2CCN(CCNC(=O)CCCF)CC2)(CC)CC1 5072,C1(CN(C(C2CCC(=O)N2)=O)CC)CCC(NC(=O)C(C2(O)CCCC2)F)CC1 5073,c1(C(=O)NC2CCCCN(C(=O)CCc3ccco3)C2)cc([N+](=O)[O-])ccc1Cl 5074,c1(C(C(=O)NCC2(OC)CCN(C(COCCC=C)=O)C2)C)cc(F)cc(F)c1 5075,c1(CCOC)nc(=NC2CCCC3CN(C(C4(CO)CCOCC4)=O)CC23)s[nH]1 5076,c1(CC)ccc(C(=O)NC2CN(C(=O)C(CC)SC)CC2(C)C)cc1C#N 5077,Cc1nc2c(N3CCCC(O)(CNC(=O)CN4CCCCC4=O)C3)ncnc2[nH]1 5078,C1(NC(Cc2c(C)n[nH]c2)=O)CC2(CCN(C(=O)C(C)C3(O)CCC3)CC2)C1 5079,C1(CNC(C(C)N(C)C)=O)CCCCN(C(=O)CN2CCCCCCC2=O)CC1 5080,CCCCC(O)C(=O)NC(CNC(=O)Cc1ccc(F)cc1CC)CC 5081,C1(CNC(C(C2CC(NC(c3cc(C)c(C)s3)=O)C2)F)=O)CC2(CC2)C(=O)O1 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5100,Cc1nn2cc[nH]c(=O)c2c1C(=O)NC1CCCN(C(=O)C(C)(C)C)CC1 5101,N1(C(C(CC)CN(C)C)=O)CC(C(N2CCCCC2CN(C)C)=O)C2(CCC2)C1 5102,Cc1nc(NC2CCCC(NC(=O)Cc3ccc(C)nc3)C2)c2scc(C)c2n1 5103,C1(NC(c2n(CC)nnc2)=O)CCC(N(C)C(c2oc(C)cc2C)=O)CC1 5104,c1(CC)cc([N+](=O)[O-])ccc1N1CCC(N(C)C(c2cc3sccc3[nH]2)=O)C1 5105,c1(NCCCCC=C)nc[nH]c(=NCc2cc(C)ncn2)c1C 5106,C=CCC(CC(F)F)NC(=O)C(F)C(C)CNC(c1ncoc1C1CC1)=O 5107,c1(C(N2CC(C)N(C(C3COC(=O)O3)=O)CC2)=O)nn(C)c2ccccc2c1=O 5108,C1(C)(CNC(C2(CC#C)CCCO2)=O)CCCN(C(=O)C=C(C)C(C)C)C1 5109,Cc1ccccc1C=CC(=O)NC(C(=O)N1CC(c2ccccc2)C1)C1CCC1 5110,N1(C(CN(C(C)=O)C)=O)CCN(C(c2cc(C)cc(C)c2)=O)C2CCCC12 5111,C1(C)(C)CCCCC(=O)N1.C1(COC)CCC(NC(=O)C=CCF)CC1 5112,c1(C(=O)NCCN(C(C2CC(C(F)(F)F)C2)=O)C2CC2)cccc2ccnn12 5113,C1(C(=O)NCC(C)(C)NC(CC=CC=C)=O)CCC(NC(=O)OC(C)(C)C)CC1 5114,CCCCC(CC)CC(=O)N1CC(F)(F)CC1CNC(=O)CCOC1CCC1 5115,CCC(C)(C)CC(=O)NC(C)CC(=O)N1CC(CC(F)(F)F)C1 5116,C(CC(=O)N(C1CC1(C)C)C)N(C(C1(CC(=O)OC)CC1)=O)CC1CC1 5117,c1(C(N2CC(C)C(NC(c3cc(Cl)cs3)=O)C2)=O)cc(N)c(F)c(F)c1Cl 5118,C1(Cl)(C(=O)NCC(C)NC(c2cnnn2C)=O)CC12CCC2 5119,c1(OC)cccc2c(SC3CNCC3C#N)ccnc12 5120,Cc1ccc(Oc2ccc(C(=O)NC3CC=CCC3)cc2)cc1C 5121,c1(C(c2nnnn2CC2CCOCC2)NCC2(CCO)CC2)cc(Cl)no1 5122,C12(C(=O)NCc3ccc(OC)cn3)CC(CN(C(=O)C(C)(C)C3(O)CCC3)C1)C2 5123,C1(C)(CNC(CN2CCN(C)CC2)=O)CN(C(C2CC(F)C2)=O)C(C)(C)C1 5124,C1(NC(C(=O)NCC2(CNC(C=CCC)=O)CCCC2)C)CCCCC1CC 5125,C1(C(N2CC(OCCNC(C#CC(C)C)=O)C2)=O)Cc2ccccc2N(C)C1=O 5126,CC(C)(C(=O)NCC1CCN1C(=O)COCCCF)C1(C)CC1(F)F 5127,O(NC(=O)C(CCOCCO)NC(=O)C(F)=C(C)C)CC=C 5128,C(CCN=c1[nH]c2c(c(=NC3CC4C=CC3CC4)[nH]1)COC2)c1n(CC)cnn1 5129,C12(NC(=O)CC3CCCO3)CCC(CNC(=O)Cn3cnnc3O)(C1)OC2 5130,N1(c2cc(NCC3CC4(CC4)CO3)nc(COC)n2)CCN2C(=O)NCC2C1 5131,C1(CC(=O)NC(COC)C(=O)NCCCC2CCCC2)COCC(C)O1 5132,N1(CC(=C)Cl)CC2CCC(NC(c3ncn(CC)n3)=O)CC2C1 5133,c1(CN2CC(C(C)NC(c3ccc(C(C)=O)cc3)=O)OCC2)cc2n(n1)CCC2 5134,C=CCC(C(=O)NCC#CCNC(=O)CCC(N)=O)c1ccccc1 5135,c1(CCCC=C)ccc(C(=O)NCC(C2CC2)NC(C2(N3CCCC3)CC2)=O)cc1 5136,C(CC(C(=O)NCCC1CCN(C)C1)NC(=O)Cn1ccc(C)c1)OC 5137,C1(C(=O)NC2CC(C)(NC(C(c3ccc(C)o3)C)=O)C2)CN(C)CCO1 5138,N1(C(C=C(COC)C)=O)CC(C)CN(C(=O)Cc2c(N)nc(C)nc2O)CC1C 5139,c1(C(=O)NC2CC(NC(c3scc(OC)c3)=O)C2)cc2c(nc1O)CCCC2=O 5140,c1(C(=O)NCC2(F)CN(C(CCC)=O)C2)ccc(F)cc1OC(C)C 5141,Cc1cc(C)c(C(N2CCCC(NS(=O)(=O)c3nccs3)CC2)=O)cc1Br 5142,n1(CCNC(C=C(C)C)=O)ccc(C(N2CCC(CC(N)=O)C2)=O)c1 5143,CCC(C)(C)C(O)C(=O)N1CCCCC1CNC(=O)C(O)CC(C)C 5144,N1(C(c2nccc(Cl)c2C)C(=O)NC(CC)C)CC(C(=O)OC)OC(C)(C)C1 5145,N1(C(c2cc(C(=O)OC)nn2C)=O)CC(OC)CC(NC(=O)CCNC(=O)OC)C1 5146,C12(CNC(=O)CC3CC=CC3)CCC1CCN2C(=O)C1=NOCC1 5147,C1(NC(CC(C=C)CC)=O)(CNC(c2nn(CC)nc2C)=O)CC2CCC1CC2 5148,N1(C(c2ccc(C(F)(F)F)cn2)=O)CC2CN(C(c3sccc3F)=O)CC12 5149,C1(NC(C(CC)=CC)=O)CC2CCC1CC2NC(=O)C(c1ccc(Cl)cc1F)O 5150,c1(C(=O)NCC(CNC(CC2CCN(C(C)C)CC2)=O)O)nsc2ccccc12 5151,C=Cc1ccc(CN2CCN(C(=O)OC(C)(C)C)C(C(F)(F)F)C2)cc1 5152,N1(C(C(C2CC(F)(F)C2)CC)=O)CCC(CON(C)C(C2CN(C(N)=O)C2)=O)CC1 5153,Cc1cc(C)nc(SCC(=O)NCC2(NC(c3csc(C#N)c3)=O)CCC2)n1 5154,c1(C(N)=O)c[nH]c(C(N2CCC(CCNC(=O)C=C3CCCC3)C2)=O)c1 5155,c1(C(N2CCC(CNC(c3cnc(Cl)[nH]3)=O)C2)=O)ccncc1N1CCCC1 5156,c1(OC)ccc(CNCc2cnc(C)c(C)c2)c(N)c1Cl 5157,C1(CNC(C2CCCO2)=O)(CO)CC12CCN(C(=O)CC(F)(F)C(F)(F)F)CC2 5158,N1(C(C(C)N(C(C)=O)C)=O)CCN(C(=O)CCCCCN(C)C)CC1CO 5159,N1(CCC)CCCC1C(=O)NC1CC(C)(NC(=O)C(c2ccc(C)s2)C)C1 5160,C1(C(=O)NC2(CNC(=O)COCc3nc[nH]n3)CC2)CCNC(=O)C1 5161,C1(NC(CC2C(C)CCO2)=O)CC2(CCN(C(c3ccoc3C3CC3)=O)CC2)C1 5162,C1(CNC(C(C2CCCC2)OC)=O)CCCN1C(C1CCS1(=O)=O)=O 5163,Cc1nn(C)c(Cl)c1C(N1CCN(C(c2coc(Cl)n2)=O)C(c2cn[nH]c2)C1)=O 5164,CC1OC(C)CC1C(=O)NCC1(NC(c2sc(N(C)C)nc2Cl)=O)CC1 5165,Cc1ccc(Cl)c(F)c1C(=O)NCC=CCNC(=O)CCSc1ccccn1 5166,c1(C(=O)NCC2N(C(Cc3ccc(C)s3)=O)CCC2C)ccc(=O)n(C)n1 5167,C1(Cl)(C(=O)NC2CC(NC(C(C)OCC)=O)C2)CC1(C)C 5168,c1(CNC(C(=O)Nc2ccc(NC(=O)OCC)c(C)c2)=O)c(C)ccc(C)c1O 5169,c1(C(=O)Nc2ccc(C)nc2Cl)ccc2c(C(N3CCC(C#N)C3)=O)n[nH]c2c1 5170,c1(OCC)ccc(Br)c(NC(C)CSc2ccccc2)c1 5171,C1(C(=O)NC(CC=C)CO)CCN(C(=O)C(C)COC)C12CC2 5172,C(C)(CCCCNC(c1cnc(OC)s1)=O)NC(c1cnc(CCCC)s1)=O 5173,Cc1ccc(-c2cccc(NC(C3CC4CCC3O4)=O)c2)cc1 5174,N1(CC(=O)N(CCC(C)NC(=O)COC(F)F)C)CCCC(N(C)C)C1 5175,S(=O)(=O)(c1cccc(N2CCCC2)n1)N(C)Cc1cc(Br)cs1.C12COCC1N2 5176,C(=O)(C1CCc2cc(F)ccc21)N1CCC(C2CC2)(NC(CC=C(C)C)=O)C1 5177,N1(C(C(C)N=[N+]=[N-])=O)CC(C)(C)CC1CC(=O)NCCC(=O)NC(C)(C)C 5178,C(=O)(C1Cc2ccc(F)cc21)N1CCC(OCCNC(c2sc(O)nc2O)=O)C1 5179,C1(N(C(CSCc2nc(C)sc2)=O)C)CCN(C(=O)Cc2cccnc2)CC1C 5180,CC(C)(CCCNC(C1CC12CC2)=O)C(=O)N1CCCC(CC2CC2)C1 5181,C(=O)(C(=O)CC(C)C)N1CC(CC=C)(NC(=O)Cc2cnsc2)C1 5182,CC(C)C(C)(CNC(=O)C(CNC(=O)C=Cc1cncn1C)N(C)C)C(C)C 5183,C1(C(=O)NCCC(C(=O)NC(C)CO)OC)CC2(CCCO2)C1 5184,C1(C(=O)N(C(C)C(C)C)C)(CC)CCCN(C(c2csc(CO)n2)=O)C1 5185,c1(C(=O)NC2CC(NC(c3nc(OC)c(F)cn3)=O)C2)ccc(C#N)cc1F 5186,C1(NC(C2C(C)CCC2)=O)CCOC12CCN(C(=O)C(C)(C)CCCO)CC2 5187,c1(CC(=O)NCC2(OC)CN(C(C3CC3(C)C)=O)C2)ccc(F)cc1C 5188,c1(C(=O)NC2C(CNC(C(COC)(F)F)=O)C2)c(Br)nc2n1CCCC2 5189,C1(OCC)CCC(CC(=O)NCCNc2cnn(-c3ccc(Cl)cc3)c2C)CC1 5190,Cc1ccc(C(=O)NC(CO)C(C)NC(=O)CC2(CO)CC2)c(N)c1Br 5191,c1(OC)cc(C(N2CCC(C3(NC(=O)CCC(C)(C)F)CC3)C2)=O)cc(N)c1O 5192,Cc1cnn(C)c1CNC(=O)C(c1cn(C)nn1)NC(=O)CCC(C)N(C)C 5193,c1(C(=O)NC2CCN(C(c3c(C)cccc3O)=O)C2)ccc2cnccc2c1 5194,C(=O)(C1CCCn2c(C)nnc21)NC(C(C)(C)NC(Cn1c(C)cc(C)n1)=O)C 5195,C1(C(=O)NCC(C(C)(C)C)NC(C=Cc2c(C)ccs2)=O)CCc2nc[nH]c2C1 5196,C(CC(C)(C)CC(=O)NCC1CCCCN(C(=O)CC2CC(=O)C2)C1)OC 5197,CC1CCC(CN(C(C2(O)CCC2)=O)C2CC2)CN1C(=O)Cn1cncn1 5198,N1(C(c2cccnc2Br)=O)CC2CN(C(c3c(Cl)cncc3Cl)=O)C2C1 5199,N1(C(CCSCC)=O)CCC(C2CC2)C1CNC(=O)C(F)=CC1CC1 5200,Cc1c(C(N2CC(C)(NC(=O)CC3CCCO3)C2)=O)oc2c(Cl)cccc12 5201,c1(C(=O)NCC(N(C)C(c2cn(C)cn2)=O)C2CC2)ccc2c(c1)NC(=O)C2 5202,CCCCS(=O)(=O)CC(=O)NCc1ccc(CNC(=O)CC#N)cc1F 5203,c1(OC)ccc(C=CC(=O)NCc2ccc(I)cc2C)cc1F 5204,C12(C(=O)NCC3(OC)CCOC3)COCC1CN(C(C1CCC1C#N)=O)C2 5205,c1(NC(CN2CCN(C(c3c(C)nc[nH]3)=O)CC2)=O)cc(Cl)cc(Cl)c1Br 5206,CON1CC(C(N2CCC(NC(C3CC=CCO3)=O)CC2)=O)CC1=O 5207,C=CCCCC(C(=O)NCCc1ccncn1)NC(C1C2CCCCCC12)=O 5208,N#Cc1cccc(C2(NC(C3CN(C(=O)C4CC4)C3)=O)CCC2)c1 5209,N1(C(c2n(C=C)ncc2)=O)CCC(C)CC1CNC(=O)CC 5210,Cc1cccn2cc(C(N3CC(CNC(=O)NC(C)(C)C)C(F)C3)=O)cc12 5211,Cc1sncc1C(=O)NC(C)C=CC(=O)N(CCS(C)(=O)=O)C 5212,c1(C(C(=O)NCCC2CC2)N(CC(C)S(N)(=O)=O)C)cccc(Br)c1OC 5213,C(=O)(CC(C)C(C)(C)C)N1CCC(F)(CNC(c2c(C)con2)=O)CC1 5214,CC1(NC(C2CCC3CCC2O3)=O)CCN(C(=O)CC2CC=CCC2)CC1 5215,C(Cn1cncn1)(C(=O)Nc1c(C(=O)NCC2(C(O)C(C)C)CC2)cc[nH]1)OC 5216,N1(C(c2ccc(CC)cc2)=O)CC(C)CCC1CNC(C1CN(CC(C)C)C1)=O 5217,c1(C(=O)NCC2(C)CCC(NC(c3cnc(COC)s3)=O)C2)cc(C)ccc1O 5218,c1(CC(=O)NCCCCCNC(C(CCC)F)=O)ccc(F)cc1C 5219,Cc1cnccc1C(N1CCCC1C(C)NC(c1cnn(CC(F)F)c1C)=O)=O 5220,C1(C(=O)OC)C(F)(F)C12CC(C(N1CCN(C(c3cnnn3C)=O)C(C)C1)=O)C2 5221,C(CC(C)C)(C(=O)NCCCCCN(C)C(C1CC12CC(C)(C)C2)=O)NC(C)=O 5222,C(=O)(C1=CC2CCCCCCC12)NC1CN(C(C2N(C=O)CCC2)=O)C1 5223,C1(C(N(CC(C)(C)CNC(C2CCCCC2F)=O)C)=O)CCC(=C(F)F)CC1 5224,c1(C(N2CC(OC)(CNC(=O)C(C)C(C)(C)C)C2)=O)ccc2ncccn12 5225,CC1OC2(C(=O)NCCCN(C(=O)CC#N)Cc3ccccc3)CC1C2 5226,CC(C)(C)CC(=O)OCC(C)(C)C.C1CC(O)CNC(=O)C=CCS1 5227,CCCC(CC)C(c1nnnn1Cc1ccco1)NCc1nnnn1C1CCC1 5228,CC1c2ccccc2OC1C(N1CC(NC(=O)COCCF)C(C)C1)=O 5229,N(C(=NCc1cccc(F)c1)NCC12CC(C1)C(C)O2)C(C)C1CC1 5230,CC(C)C#CC(=O)NCC1CCCN(C(=O)CCCc2ccccn2)C1 5231,N1(C(C2C(OC)C2)=O)CCC2CN(C(c3cnn(C)c(=O)c3)=O)CCC12 5232,c12cccc(OC)c1ONC2.n1(CC)cnc(CC(Oc2cccnc2)OC)c1 5233,CN1CCC(C(=O)NC2CCN(C(c3oc(C(F)(F)F)nc3C(F)F)=O)C2)CC1 5234,C1(C(=O)NCC(C(C)O)O)CCC2(CC2)N1C(c1cccc(CO)n1)=O 5235,c1(C(=O)NCC2CCN(C(=O)CC3CCSC3)CC2)ccnc2ccnn12 5236,C1(CNC(C2C(C)(C)C2)=O)(CNC(C2CC(n3cnnc3)C2)=O)CC12CCC2 5237,C1(CNC(CC(C)(C)SC)=O)CCC(C)N(C(c2ccc(F)o2)=O)C1 5238,C(=O)(CC(C)CC(C)(C)C)NCC(CC)(CC)NC(c1cc(C)c(O)c(C)c1)=O 5239,CCC(C)(C)C(O)C(=O)NC1CN(C(c2cc(Cl)cc(C)c2O)=O)CC1OC 5240,C1(C(=O)NC(c2ccoc2)C)CC=CCN1C(c1cccc(CO)c1)=O 5241,c1(OC)ncc(C(=O)NC2(C)CCCN(C(C3CN4CCC3CC4)=O)C2)cc1F 5242,N1(C(C(CC)OCC)=O)CC2(CCN(C(=O)C(CC)C(C)(F)F)CC2)C1 5243,CC1SCCC1NC(c1ccc(CNC(=O)Cn2cnc(=N)[nH]2)s1)=O 5244,c1(NC(CNC(c2cn(C)nc2C(F)F)=O)(C)C)ccccc1[N+](=O)[O-] 5245,N1(C(C(C(=C)Cl)(C)C)=O)CCC2CN(C(c3ccn4nncc4c3)=O)CCC2C1 5246,N1(C(C(CC)C)=O)CC2CCOC2(CNC(c2cc(CC3CC3)cc(C)c2)=O)C1 5247,N1(C(C(C(=C)C)(C)O)=O)CCC2(CC1)CC(CNC(=O)CCC(C)C)C2 5248,c1(C(=O)Nc2scc(C(=O)NCCNC(C)=O)n2)c(O)ccc(F)c1F 5249,C(=O)(C(CC(C)C)NC(c1c(C)cnn1C)=O)NC(CC)COCC1CC1 5250,Nc1ccccc1OCC1(O)CCNC1.C1C(=O)O1 5251,S(=O)(=O)(c1cc([N+](=O)[O-])c(N)cc1Cl)N1CCC(N2C(C)(COC)COCC2)CC1 5252,C1(NC(C=C(CCN(C)C)Cl)=O)CN(C(c2ccncc2N(C)C)=O)C(C)(C)C1 5253,C1(NC(CN(CCC)C)=O)COCCN(C(=O)C(c2cccc(C#N)c2)(C)C)C1 5254,Cc1c(C(=O)NC2CC(NC(=O)CCN3CCCC3)C(O)C2)c[nH]c1C#N 5255,N1(C(C2CCCCCCN2C(C2CCC3CC2CO3)=O)=O)CC2(CCOCC2)C1 5256,CC1CC(C(=O)NCCC2CCCCC2O)N(C(c2ncncc2Cl)=O)C1 5257,C(C(CC)(CC)NC(=O)Cc1ncc(C)s1)NC(C(CC)F)=O 5258,C1(CC=C)(NC(c2sccc2Cl)=O)CC2CCC(C1)N2C(C1C=C1C)=O 5259,C(=O)(CC(C)CC(=O)NCC(O)C(=O)NC1CC(C(C)O)C1)OC 5260,C1(NC(Cc2nc(COC)sc2)=O)CC(NC(c2cc(C)cs2)=O)C(O)C1 5261,C1(CC=C)(NC(c2cnc(O)cc2O)=O)CC2CCC(C1)N2C(=O)C(C)(C)CF 5262,C(=O)(CS(=O)(=O)CC(C)C)NC1CCC(CNC(C(CC(C)=O)(C)C)=O)C1 5263,CC1CCN(C(=O)CCn2ccnn2)C(CNC(C2CCCS(=O)(=O)N2)=O)C1 5264,c1(OC)nc(Cl)ccc1C(N1CC2C(NC(=O)C=Cc3cnccc3C)C2C1)=O 5265,N1(C(c2ccc(CSC)cc2)=O)CCC2(CNC(C3CC3(C)C)=O)CCCC12 5266,C1(CNC(Cc2ccc(OC)cn2)=O)CC12CCN(C(=O)C(C)(O)C(C)C)CC2 5267,C(CCCC(=O)N(C)CC1CCC(=O)N1)N(C(=O)Cn1cnc(C#N)n1)C 5268,CCC(C)(C)C(C)(O)c1nc(Cc2ccsc2)no1 5269,c1(C(N2CCN(CC(C)O)CC2)C(=O)NCCC2CC2)ccc(C2CC2)c(F)c1 5270,C(=O)(C(C)CC(N)=O)N1CC(O)(CNC(C(C)Oc2cccc(N)c2)=O)C1 5271,C1(NC(COCCCCC)=O)C(C)(C)CN(C(=O)C(C)CC(C)CC)CC1(C)C 5272,N(C1c2ccccc2CC12CCOCC2)Cc1cccc(NS(=O)(=O)C2CC2)c1 5273,N1(C(CC(C=C)C)=O)CCC(C(=O)NC(c2nc(=O)o[nH]2)C)C1(C)C 5274,N1(C(=O)Cc2ccccc2F)CC2CC(C1)N2C(c1cc(F)ccc1I)=O 5275,c1(C(=O)NCC2CC(F)(CNC(C3CCC(C)O3)=O)C2)cnc(O)c2ccsc12 5276,c1(C(N(C2CCCN(C(C3CCS3(=O)=O)=O)C2)CC)=O)ccnc2c1nnn2C 5277,c1(CS(=O)(=O)NCc2c(N3CCN(C)CC3)nccc2)ccc2c(n1)OCCO2 5278,C1(C2CC2)(CNC(CCC(C)(F)F)=O)CCN(C(c2cncc3ccsc23)=O)C1 5279,c1(CC)cnn(CC(=O)NCCCN2CCC(NC(C3CCC4CC34)=O)C2)c1 5280,C(=O)(C(C(C)CC)NC(=O)C(C#N)C(C)C)NCC=CC 5281,Cc1nn(C)c(Cl)c1CN1CCCC1CNC(c1cc(C(C)C)nn1C)=O 5282,CCC1=C(C(=O)NCC2CC(CNC(c3cc4cscc4s3)=O)CO2)CCCO1 5283,N1(C(CCC=C(C)C)=O)CC(CN(C(=O)C(O)C(C)(C)C)C)C2(CC2)C1 5284,CCC(CCc1ccccc1)C(=O)N1CCCC(c2ccc(C)cc2)CC1 5285,c1(C(N2CCC(F)(C(N3C(C(=O)OC)CC3)=O)C2)=O)ccc(C)nc1OC 5286,CC1CC(NC(=O)C(CCOCCO)NC(c2ccncc2)=O)CC(C)C1 5287,CC1CC(C)CN(c2nnc(-c3cc(F)ccc3Cl)n2Cc2n[nH]cc2Br)C1 5288,N1(C(COCCC(C)C)=O)CC2CC(C1)C2NC(c1ncoc1C1CCC1)=O 5289,c1(C(=O)NCC(C(C)(C)C)NC(c2ccc(C)n2C)=O)cc2n(c1)CCOC2 5290,c1(OC)ccnc(CNC(=O)CC2CC(C)N(C(c3sccc3CO)=O)C2)c1 5291,C1(C(=O)O)CCN(C2CC2)CC1.C12CCC(C3CCC3)N1C2=O 5292,c1(C(c2n(CCCSC)nnn2)NCc2cccc(Cl)c2)c(F)ccc(Br)c1Cl 5293,C1(C(C)(C)CO)CCCN1C(=O)C(O)CNC(=O)C(C1CC(F)(F)C1)(CCl)c1ccccc1 5294,C1(CNC(C2C(C=C(C)C)C2C)=O)(NC(c2nn[nH]c2Cl)=O)CCCCC1 5295,c1(C(=O)NC2CCCCN(C(C3(C)CCCOC3)=O)C2)ncnc2cc[nH]c12 5296,c1(SC)cccc(NC(N2CCCC2C2CCCN(C(C3CCCC3)=O)C2)=O)c1 5297,c1(C(c2ccccc2)NC2(C(F)F)CCOC2)ccccc1.CC1COC(=O)N1 5298,c1(C(=O)NCCCCNC(C2(CC#C)CCOC2)=O)cc(-n2ccnc2)ccn1 5299,O=C(C1=CCCC1)NCC1CCCN1C(=O)CCc1cnc(C2CCC2)o1 5300,CC1CN(C)CC(C(=O)NCC(C)(C)CNC(=O)COc2cccc(O)c2)O1 5301,c1(CC(=O)NCCN(C(C2CC(O)C2)=O)C2CC2)cccc2[nH]ncc12 5302,c1(C(=O)NC(CC)CNC(=O)C=C(C)C)c(Br)ccc(OC)c1C 5303,Cc1cccc(C2(NC(=O)NC3CCCCC3N3CCOCC3)CC2)c1I 5304,N(C(=NCc1cc(CN2CCCC2)on1)N1CCC(COC)C1)C(C=C)C 5305,C1(C)(C(=O)NC(CCCC)CNC(C2(C)CCCC2(F)F)=O)CCC(C)(C)CC1 5306,N1(C(C(C)CN(C)C)=O)CC(CC(=O)N(C)CCC2CCOCC2)C(C)C1 5307,CC1CN(S(=O)(=O)N2CCCC(N3CCCC3)CC2C)CCN1 5308,N1(C(C(c2ccc(OC)nc2)OC2CCCC(=O)N2)=O)CC2(C1)CN(C(C)=O)C2 5309,c1(C(c2ccncc2)N(C(=O)CC2CC3CCC2C3)C)ccc(Cl)cc1 5310,c1(CC)cccc(C)c1C(N1CCN(C)C(CNC(C2CC(OC)C2)=O)C1)=O 5311,c1(OC)cc(CC(=O)NCC(C)(C)CNC(c2c[nH]c(=N)cc2C)=O)ccc1F 5312,Cc1cnc(C#N)nc1N(C)CCN(C)C(C1COCCO1)=O 5313,CC(C)(C)C(CNC(C1CCC(F)(F)C1)=O)NC(c1ncccc1Br)=O 5314,c1(C(=O)NCC=CCNC(c2cnc(CC(C)C)s2)=O)ccc(Br)nc1O 5315,C(=O)(CC(F)(F)Br)NCC1(COC)CN(C(C2CCN(C)C2=O)=O)C1 5316,C(=O)(C1=CCC(C)(C)CC1)N1C(CNC(c2c(C)oc(C)c2C)=O)CC(F)(F)C1 5317,C1(C(=O)NC2CCN(C(=O)C(O)C3CCC3)CC2)CCCc2ccccc2C1 5318,Cc1cnc(C(=O)NCCCCC2CCCC2)c(S(=O)(=O)N2CCC(CF)C2)c1 5319,CC1(C)COCCC1CCNS(N)(=O)=O.N12CC3(CC3)CC1CC(=O)NC2=O 5320,C(C#Cc1cccnc1)NC(C(CCOCC)NC(C1CN(C)CCN1C)=O)=O 5321,N1(C(C2CC(C)(F)C2)=O)CCCC12CCCN(C(c1cccc3c1CCN3)=O)C2 5322,N1(C(CNS(CC)(=O)=O)=O)CCN(C(c2ccnn2CCF)=O)C(C(F)F)C1 5323,C1(C(=O)NC(CC2CN(C(CC=CCOC)=O)C2)C)Cc2cccc(F)c2O1 5324,c1(C(N2CCC(C)(CNC(=O)Cc3ccoc3)CC2)=O)ccc2nc[nH]c2n1 5325,c1(C(N(C2CCN(C(=O)CC3(OC)CC3)C2)CCC)=O)ccnc(C(C)(F)F)c1 5326,c1(C(N(CCN(C(=O)CN2C(=O)CCC2=O)CC)CC)=O)cccc(C2CC2)c1 5327,C1(CSc2nccc(NC(C3CS(=O)C3)=O)c2)CC12CCCOC2 5328,CCC(CC(C)C)C(=O)NCCC1(NC(=O)CC(C)n2cccn2)CCCC1 5329,Cc1nc2n(c1CC(N1CC(NC(=O)CC3CCC(C(N)=O)C3)C1)=O)CCCC2 5330,n1(C(C)C)cc(C(=O)NCC(C)NC(C2CCN(c3nccn3C)C2)=O)cn1 5331,C1(NC(=O)CCN2CCC(F)C2)CCC2CN(CCC3CCCCC3)CC2C1 5332,c1(CN2CC3N(S(C4(CC=C)CC4)(=O)=O)C(C3)C2)cc(OC)c(O)c(I)c1 5333,N1(C(CN(C2CCCC2)C)=O)CCC1CNC(C1CC(n2ccnc2)C1)=O 5334,c1(C(=O)NCC23N(C(CC(=C)C)=O)CCC2CC3)noc2c1CC(C)(C)CC2 5335,CCC(C)C(=O)C(=O)N1CCC1C(=O)NC1CC=C(C)CC1 5336,C(=O)(C(C)C(O)CC(C)C)N1CC(F)(C(=O)NC(CCC=C)(C)C)C1 5337,CCCCCCC(F)C(=O)NC(CNC(c1cnccc1Cl)=O)C(C)C 5338,c1(OCCC)ccc(Cl)cc1NC(C1CCN1Cc1cccnc1NC(C)=O)=O 5339,C=CCC(CNC(C1CC(CC)(CC)C1)=O)C(=O)NCC1CC12CCC2 5340,c1(C(C)=O)csc(C(=O)NCC(C)(C)CN(C(=O)C(F)(F)c2ccncc2)C)c1 5341,N1(C(CCCC#C)=O)CC(C)N(C(c2ccc(C3(C)CC3)cc2)=O)CC1C 5342,N1(C(C)=O)CCC(c2nc(CC(C)C(C)(C)C)n(C3CCS(=O)(=O)C3)n2)CC1 5343,C#CCC(CC(=O)OC)NC(C1CCCCC1NC(=O)C(CCC)NC(C)=O)=O 5344,C1(C(N2CC(n3ccnc3)C2)=O)(CC)CCN(C(c2n[nH]c(C)c2Cl)=O)C1 5345,Cc1cnc(C(N2CCC(CNC(C3CC3(Cl)Cl)=O)CC2)=O)cc1C#N 5346,C1(C(N(CCC#C)CCO)=O)CN(C(c2ccc(F)c(C)c2)=O)C(C)(C)C1 5347,Cc1cc(C(C)NC2CCN(C(=O)OC)C2)cc(C)c1F 5348,c1(C(N2CC3CC(CNC(c4n(C)c(S)nn4)=O)C3C2)=O)cc2cccnc2[nH]1 5349,c1(CC(=O)N(C)CCNC(c2ccoc2)=O)csc2nccn12 5350,c1(C(=O)NCC2(C(C)NC(C3CC3C(F)F)=O)CC2)cnc2ccccn12 5351,Cc1nn(CCO)cc1C(=O)NCC(O)CNC(C1(C(C)C)CNC(=O)C1)=O 5352,c1(N2CC(CNC(C(C)C3CC3)=O)OCCC2)c(Br)cncc1[N+](=O)[O-] 5353,c1(C(N(C)CC2N(C(C3(COC)CCOC3)=O)CCC2)=O)ncccc1Br 5354,c1(C(=O)NC2C(NC(=O)Cc3ncncc3Cl)CC2)cn2ccccc2n1 5355,CC(CNC(=O)C(C)(C)C1CCC1)C(F)C(=O)NC1(C(=O)N(C)OC)CC1 5356,c1(OC)cc(C)ccc1C(N1CCNC(=O)C1c1cccc(Br)c1)=O 5357,C1(C(N2C(C(N3CCC(OC(C)C)CC3)=O)CC(=O)C2)=O)CC2(CCO1)CC2 5358,C(=O)(C(O)CC(=O)OC(C)(C)C)N(C1CCCN(C(c2cc(Cl)no2)=O)C1)CC 5359,C1(F)(CNC(C(C)(C)F)=O)CCN(C(C2(c3cccnc3)CCC2)=O)C1 5360,c1(N2CC3(CCN(C(c4c(CC)nco4)=O)C3)C2)nccc2c1C(=O)OC2(C)C 5361,c1(C(=O)NC2CC(CNC(Cc3ccc(C)nc3)=O)C2)cc2cc(F)ccc2o1 5362,C1(C(=O)NC(C2CCN(C(c3ccccc3)=O)C2)C)CCCOC1 5363,C(=O)(C1c2ccccc2C2CC1C2)N1C(c2c(OC)cccc2)CNCC1 5364,N1(C(c2c(C(C)=O)cco2)=O)CCC2(CCN(C(c3c(Cl)nn(C)c3C)=O)C2)C1 5365,CCCCCC(CC)C(=O)NC1(C)CCN(c2cc(O)nc(COC)n2)C1 5366,c1(C(N(C2CCCN(C(C34CC(F)C3C4)=O)C2)CC)=O)noc2c1CCCCC2 5367,CC1CC(C(=O)NCc2cn(C)cc2C(F)(F)F)CCC1C 5368,C1(C(N2CCCC(CNC(c3ccc(C)cn3)=O)CC2)=O)Cc2cccnc2C1 5369,C1(C(=O)NC(CC(=O)NC)C)(COC)CCN(C(=O)C=Cc2cocn2)C1 5370,C(C1=CCCCC1)(c1nnnn1C(C)(C)CC)NCCOC(c1ccccc1)CC 5371,C1(F)(CNC(c2noc3ncccc23)=O)CC2CCC(C1)N2C(c1cnco1)=O 5372,C(=O)(C(F)C(C)C)NC(C(=O)NC(CN(CC)CC)C)C1CCCC1 5373,CC(C(C(=O)O)NC(=O)OC(C)(C)C)c1ccccc1.c12nc(no1)C2 5374,C1(N(C2CCCC2)C(c2ccc(OC)cc2)=O)CCNCC12CC2 5375,C(CCCCO)N(C)C(c1cc(CNC(=O)C(c2cccn2C)=O)cs1)=O 5376,C1(NC(C2CCCC3CCCN23)=O)CN(c2nnc(C(F)F)o2)CC2(CC2)C1 5377,C1(CNC(c2c(C(C)C)ncnc2)=O)CCCCN(C(C2COC(=O)N2C)=O)C1 5378,N1(C(C2C(OCC)C2)=O)CCN(C(=O)C(C)(C)CNC(C)=O)CC(C)(F)C1 5379,c1(CN(C)C(c2cc[nH]c2N(C(C(=O)OCC)C)C(C)C(=O)O)=O)ccccc1CC 5380,N1(C(C(C)(C)C2CCN(C(C3CC34CCC4)=O)C2)=O)CC2CC2(CO)C1 5381,CC1CC(NCc2cccc(F)c2)CN(C(c2ccc([N+](=O)[O-])o2)=O)C1 5382,c1(C(=O)NCC2N(C(CN(C)CC)=O)CC(O)C2O)cccc2nc(O)ccc12 5383,n1(CC(OC)OC)cc(C(=O)NC2CCC(CNC(c3ccc(SC)o3)=O)C2)nn1 5384,CC(F)(F)CC(=O)NC(C1CCCN1C(c1ncccc1Cl)=O)(C)C 5385,N1(C(C(C)N(C)C)=O)CC(O)CC1CNC(C1CCC(CC(=O)N(C)C)CC1)=O 5386,Cc1cnc2n1CCC(C(=O)NC1CCC(NC(=O)Cc3cnn(C)c3)CC1)C2 5387,c1(NC(c2c(Br)cn(C)n2)=O)ccc(OCCNC(N2CCCC2)=O)cc1Cl 5388,c1(CC)cc(C(=O)NCC2CCN2C(c2c(NC(C)=O)c[nH]c2C)=O)cc(O)n1 5389,CCCCC(C(=O)NC(CCc1ccccc1)C(C)NC(=O)CC)NC(N)=O 5390,c1(CC(=O)NCC2(CC(=O)N(CC#C)C(C)C)CC2)cncnc1 5391,N1(C(C(CCC)NC(C)=O)=O)CCN(C(C2CN3CCN2CC3)=O)C(C(C)C)C1 5392,C1(CCC)CCCN(C(c2ccc(CNC(c3ccoc3)=O)o2)=O)CC1 5393,N1(CC(=O)NC2CCC(CCC(=O)N3CC(SC(F)F)C3)C2)CCNC(=O)C1 5394,Cc1cccc(CC(=O)NCC(C2CCC2)NC(c2cc(O)ncn2)=O)c1 5395,CC1(C)CCC2(CCCN2C(c2ccc(S(=O)C(F)(F)F)cc2)=O)CC1 5396,C1(NC(CC(=O)OC)=O)CN(C(=O)CSc2c(C)n[nH]c2C)CC1O 5397,c1(NC(C2C3C(NC(C(CC)=CC)=O)C4C(C3)C42)=O)c[nH]c2ncccc12 5398,n1(CC)ncn(NC(=O)CN(C(=O)C(CC(C)C)NC(N)=O)C2CC2)c1=O 5399,N1(C(C2CC(=C)C2)=O)CC(OC)CC1CNC(=O)C(C)CC1CCCCC1 5400,CCC(C)C(C)C(=O)NCC1(C)CCN(C(=O)CCc2ncc(C)[nH]2)C1 5401,N1(C(C2N(C(c3csnn3)=O)CCC(=C)C2)=O)CCN2CCCCC2C1 5402,CCCCC(C(=O)N1CC2(NC(=O)Cc3nsc4ccccc34)CC1C2)C(C)C 5403,CN=c1cc(C(=O)NCC23CC(NC(C4CCOC4C)=O)(CO2)C3)cc[nH]1 5404,c1(OCC=C)cccnc1C(=O)N(CCNC(=O)COCC(F)F)C1CC1 5405,c1(C(=O)NCC2OCCN(C(c3c(C)ccs3)=O)C2)ccc(N)c(F)n1 5406,Nc1c(C(N2CC=CC2CNC(=O)C(c2ccc(F)cc2)F)=O)nc(O)nc1O 5407,C1(O)(C(N2CCCC(CCNC(CCC=C)=O)C2)=O)CCCC(C)(C)C1 5408,C(=O)(C1CCc2c[nH]nc21)NCC1(C)CC(NC(C2CC3(CCC3=O)C2)=O)C1 5409,C1(NC(Cn2cc(-c3cc(N)cc(F)c3)nn2)=O)CCc2nncn2C1 5410,Cc1nc2ccc(C(N3CCCC3C(C)(C)CNC(=O)CCC3CC3)=O)cc2o1 5411,C1(NC(C2C(C=C)C2)=O)COC2(C1)CN(C(=O)Cc1cncc(O)c1)C2 5412,c1(C(N2CC(NC(C3(COC)CC3)=O)C(OC)C2)=O)ccc(O)c(C(C)C)c1 5413,Cc1ccc(C=CC(=O)NCC(N2CC(C)C(C)C2C)=O)cc1 5414,CCCCC(C)CCC(=O)NC1(CO)CCCN(C(=O)Cc2c(C)n[nH]c2C)C1 5415,c1(N(c2cc(C3CC3)ncn2)C(CCc2c(C)n[nH]c2C)=O)ccc(N)cc1F 5416,CCC(C)CC(C)C(=O)N1CCCC(NC(=O)CN2Cc3ccccc3C2)C1C 5417,C1(N(C(=O)CCc2ncc[nH]2)C)CCCCN(C(c2c[nH]c(Br)c2)=O)C1 5418,c1(C(C)=O)cc(C(=O)NCC2CCC(NC(=O)COC3CCOC3)C2)cs1 5419,C=CCN=C(NCCC1CC1(Cl)Cl)N1CCC(n2cccc2)CC1 5420,N1(C(Cn2ncc(C#C)c2)=O)CCC(C(=O)NC(c2ncc(C)o2)C)CC1C 5421,N1(C(c2c(CC)cncc2)=O)CC(C(N2CC(C(N)=O)C2)=O)C(F)(F)C1 5422,N1(CC(C(=O)C(F)CC2CCOCC2)=O)CCCN(c2nnc(COCCO)s2)CC1.O 5423,C1(CN(C(=O)C2=CC(C)(C)C2)C)CN(C(c2cc(Cl)c(Cl)n2C)=O)CC12CC2 5424,S(=O)(=O)(c1ccc2c(c1)OCCO2)NCCC(=O)OCc1ccc(SC)cc1 5425,c1(C(=O)NCC(C(C)C)NC(c2cn(C)cn2)=O)cccc2nncn12 5426,N(C1CCc2ccc(Br)cc21)C(C(N1CCCC(CCC(C)O)C1)=O)=O 5427,N1(C(CC(COC)C)=O)CC2CCCC(CNC(=O)Cn3nnc(C)n3)(C2)C1 5428,C(=O)(CC(C)(O)C(F)(F)F)NCC1(CNC(C=C(C)c2cccs2)=O)CC1 5429,c1(NC(c2cccc(NCc3cncc(C)n3)c2)=O)ccc(Br)c(Cl)c1F 5430,c1(C(=O)NC(C)C(C)NC(c2cncc(C(N)=O)c2)=O)cnc(N(C)C)c(Cl)c1 5431,c12ccc(c(F)c1)C(=O)N1C(C)CC1C(=O)N2.C1(C)(CO)CCN(C)CC1 5432,C1(C(N2CC(c3ccco3)C2)=O)CC2CCC1N2C(=O)C(O)CC1CCCC1 5433,CCCCC(C(=O)NC1CCC(NC(c2ccc(F)cn2)=O)C1)C(C)C 5434,C1(CCNC(CCOCC#C)=O)CC(F)(F)CN1C(=O)C(CC)NC(N)=O 5435,CCC(C)CC(C(=O)NCc1cncc(F)c1)NC(C1CC(=O)C1)=O 5436,C(=O)(CC(C)(C)CNC(=O)C(N1CCNC1=O)C)N(C1C(C)CCC1)C 5437,N1(C(c2ccc(OC)o2)=O)CC(NC(c2ncoc2-c2cc(C)no2)=O)C(C)C1 5438,C1(F)(CNC(C(C)OCC)=O)CCCN(C(C2(CO)CC(C)(C)C2)=O)CC1 5439,C1(NCCCC(=O)NC(C2CCC3(CC3)C2)=O)CC(O)CN(C(=O)C2CC2)C1 5440,C1(C(=O)NCC(CCNC(=O)C=CCF)OC)CCc2nn[nH]c2C1 5441,CC12CC(C(=O)NC3CN(C(C4(O)CCSCC4)=O)CC34CCC4)(C1)C(C)(C)O2 5442,N1(C(C(CC=C)(C)C)=O)CC2(CCN(C(C3C=CCS3)=O)C2)C1 5443,C1(NC(C2C(CCC)C2)=O)CC2(C1)CC2NC(=O)COCc1nc[nH]n1 5444,N1(C(=O)NCc2snc(C)n2)CCC(=Cc2cccnc2)CC1 5445,CC1CCN(C(=O)C(C)Sc2ccc(Cl)cc2Cl)CCN1C(C1CC1C)=O 5446,CC(C)C(C)C(=O)OC(C)(C)C.N12CC(C(c3ccnn3C)C1)NC(=O)C2 5447,C(=O)(CN=c1[nH]c(C)cs1)N(CCC1N(C(C2CN(C(C)=O)C2)=O)CCCC1)C 5448,CCC(CC)C(C)C(=O)N1CCN(C(=O)C(=O)NCC2CC2)CC1CC 5449,CC12CCC(C(=O)NC3CC(O)CN(C(c4cc(O)cc(O)n4)=O)C3)(CC1)CO2 5450,C(=O)(CC1=CSC2=NCCN12)NCCCC(C)NC(C1COC(=O)C1)=O 5451,N1(C(c2ccnc(C)n2)=O)CC2CCN(C(c3ccoc3C(F)(F)F)=O)CC2C1 5452,c1(C(N2C(CN(C(CCOC)=O)C)COCC2)=O)cccc(Cl)c1C(F)F 5453,C1(NC(CC2N(C)CCCC2)=O)CCC2CN(C(C3CC3(C)C(F)F)=O)CC2C1 5454,c1(COC(C2N(c3nnc(C)s3)CCCC2)=O)ccc2c(c1)C(=O)NC2=O 5455,CC1(C#CC(=O)N2CCC(CCNC(=O)CC3CCC3)C2)CCCO1 5456,c1(COC)nc2ccccn2c1C(=O)NCC(C)NC(C1(C#N)CCOC1)=O 5457,c1(C(=O)NC2(N(C(=O)CC(C=C)CCC)C)CCC2)cc2c(cnn2C)nc1C 5458,C1(NC(CCC=C)=O)CCSC12CN(C(=O)CC1CCCCCC1)C2 5459,C1(CCNC(C=CSC)=O)CCCN(C(c2ncsc2-c2ccccc2)=O)C1 5460,CCCS(=O)(=O)c1ccccc1S(=O)(=O)CCNC(=O)NC1(C(=O)OC)CC1C 5461,c1(C(=O)OC)cn(C)nc1C(=O)N(C(C)CNC(=O)C(C(C)C)OCC(C)C)C 5462,C#Cc1ccc(CNC(=O)Nc2c(C)nn(C)c2SC)nc1 5463,C1(C(=O)NC2(CC=C)CN(C(C3(C#N)CC(C)C3)=O)C2)CS(=O)(=O)CC12CC2 5464,CCN=C(NCC12CC(CCO1)C2)NC1CCCC(SC)C1 5465,c1(NC(C)(C)C)ccc(S(C)(=O)=O)c(OCC(=O)NC(C2CCCO2)CC)c1 5466,N1(C(CNC(COCCCN(C)C)=O)=O)CC(=O)NC1=O.C1(OC)CCN1C(=O)C 5467,N1(C(C2C(C)OCCC2)=O)CC2(CCN(C(c3nc4c(s3)CCCC4)=O)CC2)C1 5468,C1(C(C)C)C(NC(C2(CO)CC2(F)F)=O)CCN1C(=O)CCN1CCCCCC1 5469,C1CCCCC1C(=O)OCC.C(=O)(C(C)CC1CCCC1)C(C(C)NCCCC)=O 5470,Cc1c(C(N2CCCC(NC(C3(C)CNC(=O)C3)=O)CC2)=O)cccc1C1CC1 5471,CC(CCCC(=O)N1CCOC(CCF)C1)NC(=O)COCCN(C)C 5472,c1(C(=O)NCCCOCCN(C(c2c(C)cco2)=O)C)cc2cc(O)ccc2[nH]1 5473,C1(C(N(CCCNC(C(C)OC)=O)CCO)=O)CC(=O)NC(=O)N1 5474,C1(NC(c2ncn(CC)c2)=O)C(C)CN(C(C2(N(C)C)CCOCC2)=O)CC1C 5475,N1(C(c2cncc(SC)c2)=O)CCC2(CC1)CC(C)N(C(c1cnsc1C)=O)C2 5476,N1(C(c2ccc(CC)nc2C)=O)CCN(C(c2ocnc2C)=O)CC12CCC2 5477,c1(CCC(=O)NCC2(F)CCN(C(C(C)C(F)F)=O)C2)ccc2cccnc2c1 5478,C(C1CN(C(=O)CN2CCSCC2)Cc2ccccc21)NC(C1(C)CC1(F)F)=O 5479,N1(C(c2c(C)ncc(C)c2)=O)CC2CCN(C(c3ccc(C)c(Cl)c3N)=O)CC12 5480,c1(N(CC(=C)C)C)nc2cc(OC)ccc2c(=NCC2(CC#N)CCC2)[nH]1 5481,c1(C(=O)NCCOC2CN(C(C3CC(O)C(F)C3)=O)C2)cc2c(cn1)OCCC2 5482,CCCS(=O)(=O)CC(=O)N1CCN(C(=O)C(CC)C(F)(F)F)CC1CC(F)F 5483,C(=O)(C(C)(C)C1CCC1)NCCN(C(=O)CCc1n[nH]c(=N)s1)CCC 5484,C1(C(N2C(CNC(c3cc(CC)[nH]n3)=O)CC(O)C2)=O)CCC(F)(F)CO1 5485,C1(CNC(c2ccc(CO)s2)=O)CCCCCN1C(=O)C(F)CC1CCC1 5486,S(=O)(=O)(c1ccc(C#N)c(NCCC2CC2(Cl)Cl)c1)NC(C=C)(C)CC 5487,c1(CC(N2CC3C(C(N4CCC(C#N)CC4)=O)C3C2)=O)ccc2c(c1)OCCO2 5488,N1(C(CN2CC(CC)C2)=O)CCCC(O)(CNC(C2CC3C=CC2O3)=O)C1 5489,CC1CCCc2c(N(CCO)Cc3cn(CCC4NC(=O)CC4(C)C)nn3)cnn21 5490,N1(C(c2cccc(C(C)=O)c2)=O)C2CCC1C(C)C(NC(c1nc(C)no1)=O)C2 5491,C(=O)(CCCS(N)(=O)=O)NCC1(C(N2CCC(CC)(CO)CC2)=O)CCCO1 5492,C(=O)(C(O)CNC(=O)CC1CC1)N(CCC)CC1CC1 5493,Cc1ccccc1CC(=O)N(CC(C)CNC(c1ccc(SC(F)(F)F)s1)=O)C 5494,C1(N(C(CCCOC)=O)C)CC2CCC(C1)N2C(=O)Cc1cccc(Cl)c1F 5495,c1(C(N2CCC(C)C(NC(c3scnc3Cl)=O)C2C)=O)cc([N+](=O)[O-])cnc1N 5496,c1(CN(C(=O)NC(C2CCCCC2)C)C)cccc2cccnc12 5497,Cc1nn(C)c2sc(C(=O)NCC3CC3NC(C3CNC(=O)CC3(C)C)=O)cc12 5498,c1(C(=O)NCC(CNC(c2c(C)con2)=O)CO)cc2c(C3CC3)cccc2[nH]1 5499,C(N=C(NCC1CCCO1)N1CCC(O)CC1)c1n(C)ncc1 5500,Cc1nnc2n1CCCC2C(=O)NC1C=CC(CNC(=O)CC2=CCCC2)C1 5501,N1(C(CCc2c(C)ncnc2O)=O)CC(C)CN(C(=O)C2=CSCCO2)CC1C 5502,C(=O)(CC(C)(C)C(=O)OC)NC1CC(C(=O)Nc2cnc(CCC)nc2)C1 5503,c1(C(C)C)cc(=NCCCCNC(=O)Cc2ccc3c(c2)CCO3)[nH]cn1 5504,C(=O)(CCCCCNC(=O)C(c1cc(C)sc1C)N(CC(=O)NC1CC1)C)OC 5505,CN1CCN(CC(=O)NCCC2(O)CCN(C(C3OCCCO3)=O)C2)CC1=O 5506,Cc1cc(F)cnc1C(=O)NC1COCCN(C(=O)CCC2(C)CC2(F)F)C1 5507,N1(C(C2C(C)(C)C2C#N)=O)CC23CCCC2(C1)CN(C(=O)CCOC1CC1)C3 5508,N1(C(C(=O)NCCOC)=O)CCCN(C(c2ccnc(OC)c2)=O)CC1C(C)C 5509,C12(CNC(C(C)N(C)C(C3CC(CC4CC4)C3)=O)=O)CCCCC1C2 5510,C(C(C(=O)NC(c1ccco1)COC)NC(C)=O)CSCC 5511,N1(C(C(CCCNC(CC(CC)O)=O)O)=O)CCC(C2CCC2)CC1 5512,N1(C(COCC)=O)CCC(CCNC(=O)CNC(=O)OCC)C(F)(F)C1 5513,C(=O)(C(F)(F)c1ccncc1)N(C1CCCC1C(=O)O)C.C12CCN(C1)C2=O 5514,c1(OC)ccc(S(=O)(=O)N2CCCC(O)C2)cc1.C(CC(=O)OC(C)(C)C)N 5515,C(=O)(C(Cl)=CCl)NCCN(C(C)C)C(c1cn(C2CCCCC2)nn1)=O 5516,C1(CNC(CC(=C)C)=O)(CO)CC12CCN(C(=O)COCP(C)(C)=O)CC2 5517,c1(C(N2CC(OCCNC(CNC(CC(C)(C)C)=O)=O)C2)=O)ccc(F)cc1Br 5518,c1(N2CCCC(CNC(C(C3CCCCCC3)C)=O)C2)ncccc1C#N 5519,N1(C(C2C(NC(c3ccc(OC)cc3)=O)C2)=O)CCc2ccccc2CC1 5520,N(C(=NCC1CCOC1)N1CCC2(C1)CC(F)(F)C2)CCC12NC(=O)C(CC1)C2 5521,c1(C(=O)NCC(CC)(C)NC(=O)CCC2CC2CC2CC2)c(OC)ccnc1F 5522,c1(C2N(C(c3ccn4ccnc4c3)C(=O)NC)CC2)cc2ccccc2n1C 5523,c1(C(=O)NCC(CC(=O)NCC2CN(C)CCO2)OC)cc([N+](=O)[O-])c[nH]1 5524,C12CCCCC1C(=O)N2.C(C)(C)(C(=O)NCCCCN(C)C(C)C)OCC 5525,c1(C(=O)NC2CC3CN(C(c4c(C)nn(C)c4)=O)CC32)cncc2nc[nH]c12 5526,N1(C(CC(=O)NCCC(C)C)=O)CC(C(F)(F)F)OC(C)C1 5527,N1(C(c2cscc2F)=O)CC2CCC1CN2C(C12CC3CC1C2C3O)=O 5528,C(=O)(C1=NOC(C)(C)C1)NCC(CNC(c1cc(CC)[nH]n1)=O)OC 5529,CCC(C)C(O)CC(=O)N(CCC(=O)NCCC1CC(=O)N(C)C1=O)C1CC1 5530,N1(C(C(C)=CC2CC2)=O)CC2CCC1C(NC(=O)CC1CC3CCC(C1)N3C)C2 5531,C=CC(C)(C)CCCNC(c1cccc(Br)c1Cl)C 5532,CC1CCN(C(=O)COCC(c2ccccc2)C)CCN1C(c1cc[nH]n1)=O 5533,C1(C(C)C)CCC(C)CC1C(=O)NCC1C(C(C)C)CCN1C(=O)CN=S(C)(C)=O 5534,C1(CNC(=O)C=Cc2ncc[nH]2)CN(C(C2(C3CCC3)CC2)=O)CCC12CCC2 5535,c1(C(N(C)Cc2cccc(N3CCCS3(=O)=O)c2)=O)cc(Cl)c(Cl)cc1O 5536,N(C1CCS(=O)(=O)c2ccc(Cl)cc21)C(=O)NC(CCCCC)C 5537,CC1CCCC(CC(=O)NCCOC2CCN(C(c3cnc(N)cn3)=O)C2)C1 5538,C1(NC(Cc2c(CC)noc2CC)=O)CN(C(c2cnnc(Cl)c2)=O)CCC1C 5539,C(CN=C(NCc1ccco1)N(C)CC1CCOC1)c1c(C)n(C)nc1 5540,N1(C(CC2CCCC(NC(CN(CC)CC)=O)C2)=O)Cc2cccc(O)c2C1 5541,c1(C(=O)NCCCN(C(=O)Cc2cc(C)ccc2F)CC)ccc(N)cc1F 5542,Cc1cc(C(=O)OCC(=O)Nc2ccc(Cl)cc2Cl)c(C)n1-c1ccccn1 5543,N1(C(CCC)C(=O)NCc2ccc(Br)cc2)CC2CC3CC2C1C3O 5544,N1(C(C2C=CCN2C(=O)CN2CSCC2=O)=O)CCC2(CCOC2=O)C1 5545,Cc1cc(C2CC2)ncc1C(=O)NC1CC(CCNC(C2(C)CCCN2C)=O)C1 5546,N1(C(c2nc(C)oc2)=O)CC2CCC1C(CNC(=O)CCCCF)C2 5547,c1(C(=O)NC2(CNC(CC3C(C)=NNC3=O)=O)CCOC2)cc(C)nc(O)n1 5548,c1(C(=O)NC(CNC(C(C)OCCCC)=O)C)cccn1C1CC1 5549,C(=O)(C(C)(C)C(F)(F)CC)NCCNC12CC(NC(CSCC)=O)(C1)C(C)O2 5550,C1(N(C)C(c2ccc(O)cn2)=O)CC2CCC(C1)N2C(=O)C1=NNC(=O)C1 5551,C1(N(C(CN(c2ccncc2)C(C(C)O)=O)=O)C)CN(C(=O)C(N)=O)CC12CC2 5552,CC1CN(C(c2csc(Cl)n2)=O)CCC1NC(C1(c2ccccc2)CCC1)=O 5553,N1(CC)CCN(CC(N2CCC3C(NC(=O)C(C)C4CCC4)C23)=O)CC1 5554,C1(C(N(c2nc(N3CCC(COC)CC3)nc(C)c2)C)=O)Cc2ccncc2C1 5555,c1(NCCOCCOCCNC(C2C(=C)CC2)=O)ccoc1CC(=O)OC 5556,C=C1CC(CC(N2CC(C)(OCC)C2)=O)(C(=O)NC(COC)CO)C1 5557,C1(NC(c2cc(OCC)n[nH]2)=O)C2CC1N(C(C1(C(F)(F)F)CC(F)C1)=O)C2 5558,C1(NC(c2c(OC)cc(O)nc2)=O)C(C)(C)C(NC(=O)C=CC(=O)N(C)C)C1(C)C 5559,c1(C(=O)NCC(CCNC(CCSCC)=O)O)ccc2cnc(C)n2c1 5560,CCC(C)(O)C(=O)N1CC(CNC(=O)C(O)Cc2cnc[nH]2)C(O)C1 5561,c1(OCC)ccc(Cl)nc1C(=O)NCC1CCCC1NC(=O)C(C)c1ccco1 5562,c1(CC(N2CC(=CC(C)(C)C)C2)=O)cncc(O)c1.N1(C(C(C)S)=O)CC(C)(C)C1 5563,C(=O)(C1CCc2c(F)cccc21)NC(c1ccc(OC)cc1Br)C 5564,c1(C(=O)NC(CC(C)NC(c2ncoc2C2CC2)=O)C)ccnc(NC(N)=O)c1 5565,c1(C(=O)NC2C(CNC(CN3CC(C)(C)C3)=O)CC2)oc2ccccc2c1Cl 5566,C1(Cn2cc(CCCCCCC)nn2)CCN(C(=O)CC(O)C2CC2)CC1(F)F 5567,c1(C(N(C(CCNC(Cc2ccn(C(C)C)n2)=O)C)C)=O)cnc2[nH]ncc2c1 5568,N1(C(C(CC)N(C)C)=O)CC2CCCC(CNC(=O)CCCN(C)C(C)C)(C2)C1 5569,C=CCCC(F)(F)C(=O)NCC1CN(C(C2CCC(C)O2)=O)CCN1C 5570,C1(NC(Cc2cccc(C(C)C)c2)=O)CC2CC1N(C(C1CC(=O)N(C)C1)=O)C2 5571,N1(C(Cn2ncc(C#C)c2)=O)CCC2CN(C(=O)CCC3CC(F)(F)C3)CCC12 5572,c1(C(=O)NCC2N(C(CCC#C)=O)CCC(C)C2)cc(OC)c2c(c1)CC(C)O2 5573,c1(CC)ccoc1C(=O)NCC(C1CC1)NC(c1ccnn1C(C)C)=O 5574,Cc1ccc(C(=O)NCC2C3CN(C(C4CC(n5cccn5)C4)=O)CC23)cc1 5575,C1(C(=O)OC)CCCN(Cc2ccc(F)cc2-c2nn[nH]n2)C1C 5576,N1(Cc2cc(OCC)c(O)cc2)Cc2[nH][nH]c(=NC(=O)c3cnn(C)c3)c2C1 5577,C1(C(F)(F)F)(NC(=O)C2CC2)CCN(C(C23CCCC2CC3)=O)CC1 5578,CC1CCC(C)CN1C(=O)CSCCNC(c1csc(O)n1)=O 5579,C(=O)(CC(CN(C)C)C(F)(F)F)N1CC(O)(C(C)NC(C=C(C)C2CC2)=O)C1 5580,C(C(CC(C)C)C(=O)NC(CC(F)F)C(=O)N1C2CCC1COC2)OC 5581,N1(C(c2cccnc2O)=O)CC2CC(C1)N2C(=O)CC(O)c1ccccc1 5582,c1(C(=O)NC2CC(C)(C)N(C(c3coc(O)n3)=O)C2)cccc2cnsc12 5583,C(CC(F)F)(C(=O)NC(C)C(O)C(F)F)NC(c1c(C)non1)=O 5584,c1(C(N2CCCC(C)(OC)C2)=O)cc2c(cc1N)CCCC2 5585,Cc1cccc(C(N2CC=CC2CNC(=O)CC2CC(c3ccccc3)C2)=O)n1 5586,n1(CCOC)ncc(C(=O)NCC2CN(C(c3sc(C)nc3C)=O)C3CC23)c1C 5587,c1(C(=O)NC2CCC(C(N3CC(C)C(C)C3C)=O)CC2)c[nH]c2ccccc12 5588,N1(C(C2N(C(=O)Cn3cc(CO)nn3)CCN(C)C2)=O)CCC12CC(C)(CO)C2 5589,N1(C(C(C#C)(C)C)=O)CCCC2CN(C(=O)CCS(=O)(=O)NC)CCC12 5590,CC(C(=O)N1CCOCC1)C(=O)N1CC(C)(NC(=O)CC(=O)NC2CC2)C1 5591,N1(C(c2ccc(OC)s2)=O)CCCCC(NC(=O)C(C)Cc2ccco2)C1 5592,N1(C(CC(C)n2cccn2)=O)CCC2(COC(CNC(c3cnns3)=O)C2)C1 5593,c1(OC)nc(NC2CS(=O)(=O)CC2NC(c2c[nH]nc2C(C)C)=O)nc(C)c1F 5594,N1(C(c2cc(COC)[nH]n2)=O)CC(C)CN(C(=O)Cc2c(C)noc2C)C(C)C1 5595,Cc1cc(NC(C2C=CCCC2)=O)ccc1NC(c1cn(CCN(C)C)nn1)=O 5596,C1(CNC(CCCC(=C)C)=O)CN(C(=O)C=C(C)C(F)F)CCC12CCOC2 5597,N1(C(c2c(OC)cncn2)=O)CC(O)CCC1C(=O)N(C)CC1(CO)CC1 5598,C(=O)(CCNC(=O)OC)NCC1C(CNC(CN(CCC)C)=O)C1 5599,C12(CNC(C(CC)=CC)=O)CC1CN(C(c1csc(CC3CC3)n1)=O)C2 5600,c1(NC(=O)NC2C(CC)OCC2)ccc(CNC(=O)C(F)(F)F)c(OC)c1 5601,c1(C(N2CC3(CCC3)C2c2ccncc2)=O)nn2c(c1Br)OCCC2 5602,C1(c2nnnn2C)(NCCC(C)S(C)(=O)=O)CCC(C2CCC2)CC1 5603,n1(CC)ncc(C(N2CC(CCn3cc(CN(C)CCOC)nn3)C2)=O)n1 5604,C(=O)(C1CCCc2nccn21)NC(CCCC)CNC(c1cc(C)oc1C)=O 5605,c1(C(=O)NC(CNC(COCC(=C)C)=O)C)c(C)c(Br)n(C)c1C 5606,C(=O)(C(C)CN(C)C(=O)C1CC1)N(C(CSC)C)C 5607,CC1CC2(CCO1)CC2C(=O)NCC1CCN(C(c2c[nH]ccc2=O)=O)CC1C 5608,N1(CC(=O)NC2C3CC4C(C3)C24)CCC(F)(C2CCN(c3ncccn3)C2)C1 5609,O=C1CCCC(c2ccccc2)(CNCCCF)N1 5610,N1(C(=O)CCC=CBr)CC2(CCN(C(C3CCC4CCC(=O)N34)=O)CC2)C1 5611,C(C(O)C(=O)NC(c1cc(C)[nH]n1)C)SCC 5612,C12(CNC(C3C(C)C3)=O)CCCC1N(C(C1CCC1(C)C)=O)CCC2 5613,c1(C(=O)NC2CC(N(C(=O)CN3CCCNS3(=O)=O)C)C2)ccc(Cl)c(N)c1Cl 5614,C1(C(=O)NCCCC(=O)N(C)Cc2ccco2)CC2C=CC1C2 5615,C1(NC(C(CC)NC(=O)C(C2CCOCC2)F)=O)CC2OC(=O)CC12 5616,C1(CC)CN(C(C2(C#N)CC(=O)C2)=O)CC1C(=O)NCCCCOC 5617,c1(SC(C)C(=O)NCC2=NOC3CNCC23)cnc2ccccc2c1 5618,C1(N(C(C=CCCC)=O)C)CCCC(NC(=O)CCn2ccnc2)C1 5619,c1(C(N2CC(=CC)C2)=O)ccnc(CNC(=O)CC(C)(C)O)c1 5620,c1(C(=O)NC(c2ccc(C(=O)OC)cc2)C)ccc2c(C3=CCOC3)n[nH]c2c1 5621,Cc1nc2nc(=S)[nH]n2c(C)c1CC(=O)NC(C)C(C)NC(=O)C(F)F 5622,C12(NC(C(C(CC)C)NC(N)=O)=O)CCC(CNC(=O)CC(F)F)(CC1)OC2 5623,N1(C(Cc2cc(C)no2)=O)CCC(NC(C2CCCOC2)=O)C(O)C1 5624,c1(CC(=O)NC2CCCC2CNC(=O)C(O)CF)ccc(C(F)(F)F)nc1 5625,c1(CNC(C(C2CCCN(C(CCSC)=O)C2)(C)C)=O)cnc(F)cc1C 5626,C(=O)(C1=C(Cl)CCC1)NC1CC(F)(CNC(c2c(NC)nccc2)=O)C1 5627,Cn1nnnc1SCCC(=O)NC1CC(F)(CNC(c2cc(CCO)on2)=O)C1 5628,CC(CC(N)=O)C(=O)N1CC(CNC(=O)C2CC2)C2(CC2)C1 5629,N1(C(c2ccc(OCC)cc2)=O)CC2(CCC2NC(c2ccc(CO)s2)=O)C1 5630,C1(NC(CC=CCC)=O)CC(C)CN(C(c2ccc(=O)n(CC(F)(F)F)c2)=O)C1 5631,N1(C(C(C)C2CCC2)=O)CCOCC(NC(c2occc2-c2cnn(C)c2)=O)C1 5632,C1(CNC(CC=CC=C)=O)C(CC)CCN1C(=O)C(F)C(C)C 5633,C1(F)(CNC(COCc2n(C)ncc2)=O)CCC(CNC(C2CCCO2)=O)CC1 5634,C(C(=O)N(C)CC1CCCC1NC(=O)COC1(C)CCCC1)(C(C)(C)C)OC 5635,C1(NC(c2c(C)onc2C2CC2)=O)CCN(C(c2ccc(N)c(Cl)n2)=O)CC1F 5636,Cc1c(C(=O)NC(C(N2CC[Si](C)(C)C2)=O)C2CCCC2)ccn1C 5637,C1(C(=O)NCCN2CCN(CCO)CC2)CCc2nnc(O)cc2C1 5638,C(=O)(C1=CC2(CCN(C(c3ncc4ccccn34)=O)C2)C1)NCC(C)CCO 5639,N1(C(c2n(C)nc(O)c2)=O)CC(NC(c2cc(O)nc(Cl)c2)=O)CC(O)C1 5640,CC1(C)CC(O)(CC(=O)NCC(C)(C2CC2)NC(C23CC(C)(CO2)C3)=O)CO1 5641,CNS(=O)(=O)N1CCC(C(=O)N(CCCN(C(=O)CCNC(=O)CO)C)C)CC1 5642,C1(C)(COC)CC(NC(=O)CCc2nc(C)c(C)o2)CN1C(=O)CCCN=[N+]=[N-] 5643,c1(N(CCOCCN(C(C2C(CCC)CCC2)=O)C)C)ncnn2c(Br)ccc12 5644,c1(CNC(C(C)(C)C)c2nnnn2C2COC2)ccc(C(F)F)cn1 5645,c1(C(N(C(c2cn(-c3cccc(OC)c3)nn2)C)C)=O)ccc(S(C)(=O)=O)nc1 5646,c1(C(N2CC(C(=O)NCC3OCCN(C)C3)OCC2)=O)cccc2ccoc12 5647,n1(CC(=O)NC(C(C)NC(c2cnc(C)[nH]2)=O)C(C)C)ccc(=O)cc1C 5648,CC(C)CC(C)CC(=O)NC1CCN(C(=O)C2=CS(=O)CCC2)CC1O 5649,c1(CCC(=O)NC23CC(NC(C4NC(=O)OCC4)=O)(C2)C3)cc2ccccc2[nH]1 5650,C(=O)(C#CC(C)(C)CNC(=O)C=C(C1CC1)C1CC1)NCC1C(C)C1 5651,c1(SCC=C)ccccc1C(N1CC(NC(=O)C(c2cccnc2)O)C(C)C1)=O 5652,C1(C(N2C(CNC(c3c(C)cnnc3O)=O)CC2)=O)Cn2c(C)nnc2CN1C 5653,C1(CNC(COC)=O)CCN(C(=O)C(C2CCOCC2)OC)C(C)C1 5654,c1(C(=O)OC(C)(C)C)cnc(NC(=O)NCC(=O)NCc2ccc(Br)s2)[nH]1 5655,Cc1ccc(NC(C2CCCC(NC(=O)Cc3ccc(Br)cc3I)C2)=O)c(I)n1 5656,c1(C(=O)NCCCN(C(=O)CCCCC#N)CCC)nccc2[nH]ccc12 5657,N1(C(c2ncc(C)s2)=O)CCc2c(Br)ccc(NC(c3ccnnc3)=O)c2C1 5658,C12(C(=O)NCC3(CO)COC3)CCCNCCC1C2 5659,CC#CCCCC(=O)NC1CC(CNC(C2CCCCO2)=O)C1 5660,C(N=c1[nH]c(N2CCC(C(C)C)C2)nc2c1CCCCC2)C1(OC)CC1 5661,C(c1ccc(F)c(F)c1)=C(C)C(=O)NC1(C)CCN(C(C2CCOCC2)=O)C1 5662,C1(NC(c2nc(C)[nH]c3nccc2-3)=O)CC2CCC1(N=c1[nH]ccnc1F)C2 5663,c1(OC)cc(C(N2CCC(NC(c3ccc(C)c(N)c3)=O)C(C)C2)=O)ccc1Cl 5664,c1(C(=O)NCC(CC)NC(C2CCC2c2nc[nH]n2)=O)nc2cccnc2s1 5665,c1(C(N(C(CNC(CC2C(C)CCO2)=O)C2CC2)C)=O)nn(C)c2c1CCCC2 5666,N1(CC(=O)NCCC(O)CNC(c2cccnc2)=O)CCOC1=O 5667,c1(CC(=O)NC2CCCCC2CNC(=O)CCCCN2CCCC2)ccc(Cl)cn1 5668,c1(C(=O)NC(CC)C(=O)NC2CC3OCCC23)ccc(C#N)c(C)n1 5669,CCN=c1[nH]c(C(N2CCCC2CCNC(=O)CN(CC)CC)=O)cs1 5670,c1(C(N2CCC(NC(C(C3CCC3)OCC)=O)C2)=O)ccc(N(C)C)cc1OC 5671,C(=O)(C(C)CC(C)C)NC(c1cnn(C)c1)C(=O)NCC(C(=O)OC)(F)F 5672,c1(C(N(C(CCNC(Cc2cccc(C)c2F)=O)C)C)=O)cc2c(o1)CCCC2 5673,C(=O)(C(Cc1cnc[nH]1)NC(=O)CC1CC1)NC(CC)C1CC1 5674,C1(C(=O)NC2CCN(Cc3nc(-c4ccccc4)no3)C2)CC2CCC1O2 5675,C(=O)(C(C#N)C(C)C)NCC(CN(C(=O)CCC1CCCO1)CC)(C)C 5676,c1(SCC)cncc(C(=O)NCCNC(C2CC(O)CN2)=O)n1 5677,c1(C(C(=O)NCCOCC)N(C)CC2CCC(C)CC2)ncc2ccccn12 5678,C(=O)(C(C)(CC)C(=O)NCc1ccc(CNC(C2CCSC2)=O)cc1)OCC 5679,c1(C(=O)NCC(C(C)C)NC(c2ccc(OC(C)C)cn2)=O)cccc2sccc12 5680,c1(OC(C(=O)N2CC(n3cc(SNC(C)C)nn3)C2)(C)C)ccc(Cl)cc1 5681,C1(NC(CC2C(=O)NC(=N)S2)=O)CC2CC(C1)N(C(=O)CCC1CCCCO1)C2 5682,N1(CC=CC(=O)NCC2CCCN2C(=O)CSCc2ccccc2)CCOCC1 5683,N1(C(C2(CC=C)CCCN2C(c2ccc(C3CC3)o2)=O)=O)CC(=O)N(C)CC1C 5684,C(CCN=C(NC(c1cccc(C)c1)C)NC1CC1C1CCOCC1)OCC 5685,N1(C(CC(C)c2cnn(C)c2)=O)C2CCC1C(NC(=O)COc1ccsc1)C2 5686,N1(C(C(C2CCCC2)OC)=O)CC=C(C(=O)NC2COCCC2O)C1 5687,c1(C(=O)NCC23C(CN(C(C(CC)SC)=O)C2)CC3)ccc2c(n1)CCC2 5688,N1(CC(=O)NC(C)(C)C=CC(=O)NC2(C(N)=O)CCC2)CCNC1=O 5689,n1(CC)ncn(NC(=O)C(Cn2cncn2)NC(=O)CC2CCOC2)c1=O 5690,N1(C(CCc2ncn(C)c2)=O)C2CCC1C(NC(=O)CCN1CCOC1=O)C2 5691,C1(OC(c2cncc(OCCC(F)(F)F)c2)=O)CC2(C1)OCCO2.C1C(O)CO1 5692,C1(O)(C(C)NC(CCn2ncc(C)c2)=O)CCN(C(c2sc(F)cc2C)=O)CC1 5693,C1(O)(CC(=O)NCCN(C)C)CCN(C(c2ccc(C#N)cc2)=O)CC1 5694,c1(CC)sc(C(N2CCC(F)(C(N)=O)C2)=O)cc1CC 5695,c1(-c2cn(CC3CCC(NC(CC(CC)C4CC4)=O)C3)nn2)cc(F)ccc1Cl 5696,C(=O)(C(C)(O)C(F)(F)F)N(CCCNC(c1c(F)ccc(CC)c1)=O)CC 5697,C(=O)(CC(O)C(C)C)NC1C(CC(N2CC3C(C(C)C)C3C2)=O)CCC1 5698,CC1(C(=O)NCC2(CNC(=O)CCF)CCC2)COC(=O)OC1 5699,c1(C2CN(CCNC(CCC#C)=O)C2)ccc([N+](=O)[O-])cc1Cl 5700,C(CC)(c1ccc(C)cc1)=CC(N1CCCC(NC(C2C(C=C)C2)=O)C1C)=O 5701,c1(C(N2C(C(N(CC(C3CCC3)OC)C)=O)CC(=O)C2)=O)cc2cccnn2c1 5702,Cc1nccc(=NCC2CCCN(C(=O)CC3(C)CCS(=O)(=O)N3)C2)[nH]1 5703,C1(CNC(C)=O)(CSC2(c3ccc(F)cc3)CC3(CC3)C2)CCCCC1 5704,Cc1cc(C(c2nnnn2C2CCCCC2)NCc2nccn2C)c(C)nn1 5705,N1(C(c2c(COC)noc2)=O)CC2CC(C1)CN(C(=O)C(C)(C)C1CCC1)C2 5706,c1(C(=O)NC(c2cnc(C)s2)C)cc(S(=O)(=O)CC2CC2)ccc1F 5707,c1(OC)ccc(CN2CCCC2C(=O)Nc2ccccn2)c(C)c1C 5708,CC(C)(C)CC(C(F)(F)F)NC(C1(c2ccccc2OC(F)(F)F)CC1)=O 5709,c1(OCC(=O)NC2CCCC2CNC(c2ccnc(O)c2)=O)ccc(Cl)cc1F 5710,Cn1cc(S(=O)(=O)NCC(=O)NC2CC(NC(=O)CC3CCCCC3O)C2)cn1 5711,C#Cc1ccc(C(=O)NC(CCC=C)C(=O)NC(C)CCC=C(C)C)nc1 5712,c1(C(=O)NC2CCN(C(c3nn(C)c(Cl)c3)=O)CC2F)c(Br)cc(F)c(F)c1F 5713,C(=O)(CCCCC(C)CC)NCCC(=C)CNC(c1csc(Cl)c1)=O 5714,CCCC(C)(CC)C(=O)NC1CCCC(NC(c2ccc(O)c(C)c2C)=O)C1 5715,N1(C(C2C(C(=O)OC)C2)=O)CCN(C(=O)COc2cccc(Cl)c2)CC1CC#N 5716,N1(C(c2cc(C)c(Cl)c(N)c2)=O)CCC2(CC1)CN(C(=O)CC1CC3CC3C1)C2 5717,C1(N(C(=O)Cc2ccncc2)C)CCCCC1N(C(=O)Cn1nnc(=N)[nH]1)C 5718,C(=O)(C1CCc2ccccc21)N1C(CN(C)C(C2CC(N=[N+]=[N-])C2)=O)CCCC1 5719,CCCCC(CC)CC(=O)N1CC2CC1CN(C(c1cn(CCCF)nn1)=O)C2 5720,CC(C(=O)NC1CC(NC(=O)COCc2nnc(S)n2C)CC1O)C(F)F 5721,CCC(CCO)NC(=O)CCC1(NC(=O)C=Cc2cc[nH]c2)CCC1 5722,C12(C(=O)NCC3N(CC)CC3)CCC(CC1)CN2C(c1ccnc(C)n1)=O 5723,CCCCC(CN=c1nc(C(C)C)[nH]s1)NC(c1n[nH]c2ccccc12)=O 5724,N1(C(c2c(SC)cc(C)cc2)=O)CC(NC(=O)C(F)CC2CCC2)C2(CCC2)C1 5725,c1(C(=O)NC2CCC(NC(c3cnc(CCC)s3)=O)C2)ccnc2c1nnn2C 5726,C1(C(=O)NCCN(C(CSCCCC)=O)CC2CC2)CNC(=O)N1C 5727,c1(OC)cccc(Br)c1C(N1CCC(O)C(C(=O)NC(CO)C(F)(F)F)C1)=O 5728,Cc1cc2ncc(C(=O)NCC3CC(C)CCN3C(C3CC3(Cl)Cl)=O)c(C)n2n1 5729,N1(C(C2CC(OC)C2)=O)CCN(C(=O)C=C2CCN(C)C2)C2CCCC2(C)C1 5730,C(C1=NOC2CN(C(=O)CC3(CC)CCOCC3)CC12)NC(c1n(CC)ncc1)=O 5731,Cc1nc(C(C)C)ccc1C(=O)N(CCNC(c1cc[nH]c1)=O)CC1CC1 5732,C(c1cc(F)c(F)c(F)c1)=CC(N1CCCN(C(C2(OC)CC2)=O)CC1C)=O 5733,CCC(C(=O)N(C)CC1(O)CN(C(C2CC(=O)N2)=O)C1)C1CCOCC1 5734,c1(NS(Cc2cn(C)nc2)(=O)=O)ccc(S(=O)(=O)NC2CC2)cc1 5735,c1(OC)ccc(C(N2CC3(CC(NC(C4CCC4OC)=O)C3)C2)=O)cc1OC 5736,c1(OC)ccc(F)cc1-c1nc(CC2CCCC2)nn1C1CCCC1O 5737,c1(C(=O)NC2CCN(C(=O)C(O)Cc3ccccn3)C2)cccc2c1CCCC2 5738,c1(C(=O)NCC2(C)CCN(C(c3ccc(O)nn3)=O)C2)ccc(C#N)c(Cl)c1 5739,N1(C(c2c(C(C)C)scn2)=O)CCC(C)(C)C(NC(=O)CC2C=CCCC2)C1 5740,CC1(C)Oc2ccc(C(N3CCC4C(CCN4C(=O)C(O)C(F)F)C3)=O)cc2O1 5741,N1(C(c2c(C)oc(Br)c2)=O)CC(NC(c2ccnn2C)=O)CC(C)C1 5742,N1(C(CC(=O)OC)=O)CCN(C(=O)Cc2cc(F)cc(F)c2)CC1CF 5743,c1(CC(=O)NCC2CC(NC(=O)C=CC(N3CCOCC3)=O)C2)cncc(O)c1 5744,C(CC(C)C(=O)NC1CCC(N(CCC)C(=O)Cn2nccn2)CC1)=CC 5745,C1(NC(C2CN(C(C)=O)C2)=O)CN(C(C2(c3ccccc3)CCC2)=O)CC1C 5746,C(CNC(=O)C=Cc1ccco1)(C(C)C(C)C)NC(c1c(C)onc1Br)=O 5747,c1(C(=O)NC2CCN(C(C(COC)OCC3CC3)=O)CC2)cccn2nccc12 5748,Cc1ncsc1C=CC(=O)NC1CC(O)(CNC(C2CNC(=O)N2)=O)C1 5749,Cc1ccc(Br)c(S(=O)(=O)NCc2nnc(CC3CC3)n2-c2cccc(O)c2)c1 5750,c1(C(N(C2CCN(C(=O)C=CBr)C2)CC)=O)cc(Cl)nnc1Cl 5751,c1(C(C)C)cccc(CNC(c2cc(CNC(C3COCC(C)O3)=O)cs2)=O)c1 5752,C(=O)(CC(C)C(=O)N1CCC(C)C(NC(=O)CC2CCCCO2)C1)OC 5753,CN1CCOC(C(=O)NC(CO)C(=O)NC(C2CCOC2)CO)C1 5754,C(CCC(CC)CC)NC(C(C(C)NC(COCCC)=O)C)=O 5755,C(=O)(C(C)(C)CC(C)C)NC(COC)CC(=O)N(C)CCC1CCCCC1 5756,C1(NC(c2ccc(C(F)F)cn2)=O)CN(C(=O)CCc2nc[nH]n2)C2(CCC2)C1 5757,N1(C(Cc2c(COC)cccc2)=O)CC(NC(C2CCOCC2)=O)CC12CCC2 5758,C1(O)(C(N(CCCCNC(CCNC(C)=O)=O)C)=O)CC1(C)C 5759,N1(C(C2CCC(CC)O2)=O)CC2(C)CN(C(C3CNC(=O)N3)=O)CC2(C)C1 5760,c1(C(=O)OC)cc(=NC2CCN(C(c3ccn(C)c(=O)c3)=O)C(C)C2)[nH]c(Cl)n1 5761,c1(C(N2CCN(C(=O)CCc3cncs3)C3CCCC23)=O)n[nH]c2ccccc12 5762,N1(C(CCCC#CC)=O)CC2CC(F)(F)CCC2(NC(=O)COCC)C1 5763,S(=O)(=O)(c1cnn(C)c1)NC(C(=O)NC(C)CCNC(=O)C(C)NC1CC1)=O 5764,c1(NC(C2N(C(CN(CC(=O)OC)C)=O)CC2)=O)ncoc1CNC1CCSC1 5765,C=CCC(C(=O)N(C)CCOCCN(C)C(C1CCCOC1C)=O)OC 5766,C(c1ccn(C)c1)=CC(=O)NC1(CCNC(C(C)OCCCC)=O)CCC1 5767,N1(C(COC2CC(NC(C3C(C)CCOC3)=O)C2)=O)CC(F)CC(F)C1 5768,c1(OC)cc(N)c(Cl)cc1C(N1CCCC1CNC(=O)C1=CC2CCC1C2)=O 5769,c1(OC(C)(C)C)cccc(C(C2CC2)OC(N2CC(CCCNC(C)=O)C2)=O)c1 5770,C(C(=O)NC1CCCCC1CNC(C1CCCN1CC(F)(F)F)=O)(C(C)C)OC 5771,C1(C(=O)O)CCCCCCN1C(c1cc(C(F)(F)F)ncc1Br)=O 5772,c1(OC)ccc(Cl)cc1NC(N1CC(c2ocnc2CNC(=O)C(C)(C)C)C1)=O 5773,C1(O)(CC(=O)NCC(CN(C(=O)CS(=O)(=O)N(C)C)C)(C)C)CCCCCC1 5774,N1(C(c2nc(CCCC)sc2)=O)CCCN(C(c2cc(C)ncn2)=O)CCC1 5775,c1(C(=O)NC2CCC(Cn3cc(C4(C)CCCC4)nn3)C2)cnn2c1CCCC2 5776,N1(C(COC(C)=O)=O)CCN(C(=O)C(F)C2CCC2)C(C2CC2)C1 5777,CCC(C(=O)N1CCN(CC(O)COc2ccccc2)CC1)C(=O)O 5778,Cc1ccc(C(C)(C)C(=O)NC(C)CCN(C)C)c(C)c1 5779,c1(CC)noc2ncc(C(=O)N(CCN(c3nnc(C)s3)C)C(C)C)cc12 5780,c1(C(N2CC(O)(C(C)NC(=O)C3=NOCC3)C2)=O)c[nH]c2cc(Br)ccc12 5781,N1(C(=O)NCCc2nc(CC)sc2)CCCN2CCCC12 5782,CC(C(C)(C)NC(=O)C=C1CCCC1)NC(=O)Cc1csc(Cl)n1 5783,C(C(COC)CC(=O)N1CC(CCNC(C2(Br)CC2(C)C)=O)C1)OC 5784,C(=O)(CC(CCC)NC(=O)C=Cc1ccncn1)NCC(=C)Br 5785,N1(C(c2ccc(OCF)cc2)=O)CC2CN(C(c3cnco3)=O)CC2C1 5786,C#Cc1ccc(NC(C2CC(C)CN(C(c3[nH]ccc3C3CC3)=O)C2)=O)c(C)c1 5787,C1(NC(C(F)=C(C)C)=O)CC2CC1CN(C(=O)C(c1c(C)noc1C)(C)C)C2 5788,c1(N2CC3CN(C(c4ccc(Cl)cc4F)=O)CC32)ncnc2[nH]ccc12 5789,Cc1cc(N2CCOC(CC(N3CCOC(O)C3)=O)C2)nc(C)n1 5790,c1(NC(=O)C(=O)NC2CC(N3CCC3)C2)ccccc1 5791,N1(C(C2CC=C(C)CC2)=O)CC2CCC(C1)N2c1ccc(C(F)(F)F)nn1 5792,C1(C2CCCCC2)(C(=O)NC2CC(NC(C3(C#N)CCOC3)=O)C2)CC1 5793,C(C(C)(C)CC(=O)N1CC2CC2(CO)C1)NC(c1nn(C)c(Cl)c1)=O 5794,N1(C(C)C)CCOC(C(=O)Nc2cnccc2C(=O)OC(C)(C)C)C1 5795,c1(OC(C)C#N)ccc(CC(=O)NCCNC(c2cc(C3CC3)ccn2)=O)cc1 5796,c1(C(N(C(C)C)CCNC(C2CC3C=CC2O3)=O)=O)ccc2occc2c1 5797,C(=O)(C(CC)CC(C)C)N1CC(C2CC2)(C(=O)NC2C(CC=C)COC2)C1 5798,c1(C(=O)NC2CC3CN(C(C(C=C=C)C)=O)C(C2)C3)n[nH]c2c(C)cccc12 5799,N1(C(c2c(C)scn2)=O)CC2OCC(NC(C3CC4(C3)CC(C)C4)=O)C2C1 5800,c1(NC)cnc(C(=O)NCC2CCCN2C(C2CCN(C)C2)=O)cn1 5801,N1(C(C(CC)(C)OC)=O)CCOCC(F)(CNC(c2nnc(C(C)(C)C)s2)=O)C1 5802,CCCCCCC(C)C(=O)NCC12CCC(C1)N(C(=O)CN1CC(=O)NC1=O)C2 5803,C1(C(N(C2CCN(C(=O)C(C)(C)C3CCC3)CC2)CCOC)=O)C2CC2C2CC12 5804,N1(C(N2C(C)(C)CCC2)=O)CCC12CCC(C)CC2 5805,C(CC(=O)NCC1(CC2CC2)CC1)(CC(C)C)NC(C=Cc1cccc(C)c1)=O 5806,C(=O)(C(C)(C)CC(C)C)N(C(CC(=O)NC(C(=O)OC)C)(C)C)C 5807,C12(NC(c3n(CC#C)ccc3)=O)CCCN(C(c3cc4n(n3)CCO4)=O)CC1C2 5808,N1(c2ncnc(N(CC(CC)C)C)c2C)CCc2c[nH]nc2C1 5809,c1(C(=O)NCCC2CCC(NC(c3cc(OC)ncc3)=O)C2)nn(C)c(C)c1Cl 5810,c1(OCC)nn(C)cc1NC(=O)C(=O)NC1C=CC(NC)C1 5811,CCCC(C)(C)C(=O)NC1CC(CCNC(=O)COCCOCCO)C1 5812,CCC(C)(F)C(=O)N(C)CCN(C)C(C1(N2CCSCC2)CCCCC1)=O 5813,C1(N(C(CS(CC)=O)=O)C)CCCC2CN(C(c3ccc(N)c(Cl)c3)=O)CC12 5814,c1(C(=O)NCC(c2ccc(Br)cc2)(C)C)ccc2c(c1)NC(=O)C2 5815,S(=O)(=O)(c1ccc(NCc2cc(C)ccc2F)nc1)N1CC=C(C)CC1 5816,C12(NC(c3c(C)ocn3)=O)CC1CN(C(=O)Cn1nc(C(F)F)cc1C(F)F)C2 5817,c1(C(=O)NCc2scc(CNC(CCC=C=C)=O)n2)cccc(F)c1C 5818,N1(C(=O)Nc2ccc(C3(C)CC3(F)F)cc2)CC(S(C)(=O)=O)CC12CCCC2 5819,Cc1cc(C(=O)NC(CNC(c2cnsn2)=O)CC(C)C)cnc1C(F)(F)F 5820,c1(C(=O)NC2C(OC)CN(C(=O)C(O)C(C)(C)C)C2)cc(S(N)(=O)=O)c[nH]1 5821,N1(C(=O)OC(C)(C)C)CC2CN(C(c3ccc(Cl)cc3N3CCCC3)=O)C2C1 5822,c1(C(N(CC(CNC(C(COC)NC(C)=O)=O)O)C)=O)sc(C(C)(C)C)nc1C 5823,CC(C)CS(=O)(=O)CC(=O)NC1CC2CC(NC(c3coc(C(F)F)c3)=O)C2C1 5824,C(CS(=O)(=O)C1=NOC(C)(C)C1)NC(c1ccc(C(F)(F)F)cc1)C(=O)OC 5825,OCCC(N=c1[nH]c(=NCc2snnc2C2CC2)[nH]c2c1CCCC2)C1CCCC1 5826,c1(C(=O)NCC#CCOC)ccc(CNC(=O)CCC2(C#N)CCC2)cn1 5827,C1(CC(=O)NC(C)C(C2CCCCC2)NC(=O)OC(C)(C)C)CCCC2CC12 5828,C(=O)(CC1=NNC(=O)C1)NC1CCC(N(C(CN(CC)CC)=O)C)C1 5829,c1(C(N(CCN(C(C=CC)=O)C(C)C)C)=O)cccc(C2CCCOC2)c1 5830,N1(C(c2ccc(C)n2C)=O)CC2CCC1CN2C(c1ccc(F)cn1)=O 5831,C1(C(C)NC(c2cc(C3CCCCC3)[nH]n2)=O)CN(C(=O)CCNC(N)=O)CCO1 5832,C12(CNC(C3(CC=C)CC=CC3)=O)CC(CO1)N(C(=O)CC1(C)CC1(F)Cl)C2 5833,Cc1cccc(OCC(N2CC(OCCCS(N)(=O)=O)C2)=O)c1 5834,c1(C(=O)OC)n[nH]c2c1CCN(CC1CCC(C(F)(F)F)O1)C2 5835,S(=O)(=O)(c1cccc(=NCc2cc[nH]c(=N)c2)[nH]1)N(CC(C)OC)CC 5836,Cc1cc(S(=O)(=O)N(C(=O)C(CN)CC(C)(C)C)C(C)C)sc1C 5837,C1(C(=O)NCCC2CN(C)C(=O)C2)CCC2(CC2)N1C(=O)Cc1ccc(O)cn1 5838,C1(NC(C2CC=C(C)CC2)=O)CCC2(CC1)CN(C(=O)CCCCCBr)C2 5839,C1(S(N)(=O)=O)(C(N(C2CCC(NC(C=C(C)Cl)=O)CC2)C)=O)CCC1 5840,c1(C(=O)NCCN(CCC)C(C2CCCOC2C)=O)ccc2nc(S)oc2c1 5841,CC(C)(F)C(C)(F)CNC(c1cccnc1CNC(=O)CCC1CCCOC1)=O 5842,C1(n2cc(CCCC)nn2)CCC(NC(C2(O)CC2)=O)CC1 5843,c1(NCC2C(C)(C)CCO2)[nH]c(=NC2CCS(=O)(=O)C2)nc2scnc12 5844,c1(C(=O)OC)ccc(C(N2CCC(NC(=O)CC(C)c3ccccc3)C2)=O)nc1 5845,O=S1(=O)CCC(CNC(=S)NC2CCC3(CC2)CC3)c2ccccc21 5846,C1(NC(COC)=O)CCCC(N(C(c2ccnc(CC3CCC3)c2)=O)CC)C1 5847,C(=O)(C(C#N)C(C)C)N1C2C(C(=O)NCC(CSC)(C)O)C(C2)C1 5848,C1(CNC(COc2cc(C)on2)=O)COCCN(C(c2cnn(C)c2Cl)=O)C1 5849,C(=O)(C1=COCCO1)NCC1(CNC(C(C(C)C)C)=O)CC1 5850,C1(NC(C2(C#C)CCC2)=O)CS(=O)(=O)CC1NC(c1cc(C(C)=O)cn1C)=O 5851,C1(NC(c2cc(C3CC3)cs2)=O)CC12CCN(C(=O)CC1CC1(Cl)Cl)C2 5852,c1(C(=O)NCC(CC)NC(c2cc(C)nn2C)=O)ccc2c(C)cc(O)nc2c1 5853,c1(C(=O)NCC2CC(C)(C)N(C(C3CCNC3=O)=O)C2)ccn2cccc2c1 5854,N1(C(C2CC=C(C)CC2)=O)CCC2CN(C(C3CCC(=O)N3)=O)C2C1 5855,n1(CC(=O)N(C)CC2CCCN(C(c3cccn3C)=O)C2)cc(Cl)c(O)nc1=O 5856,C1(C(N(C2COC(C)(C)C2)C)=O)CN(C(=O)Cn2cncn2)CC12CC2 5857,c1(C(=O)NCC(C)(C)NC(c2ccc(N)cn2)=O)ncc2cc(Br)ccc2n1 5858,CCC(C)C(O)C(=O)NCC1CC(C)(C)CN1C(C1CC1(F)F)=O 5859,C(=O)(CC(CCCC)NC(=O)Cn1nccc1C)N1C(C#C)COCC1 5860,c1(C(=O)NC(C)(C)CNC(=O)CC#N)cccn2nncc12 5861,Cc1c(F)ccc(C(=O)NCC2(C)CCN(C(C3(C)CC4(CCC4)C3)=O)C2)c1C 5862,c1(CNC(c2ccc(-c3ccoc3)cc2)=O)coc2ccccc12 5863,C12(NC(CCC=C)=O)CCOCC1CN(C(=O)Cc1ccc(C)c(C)c1)C2 5864,c1(Cc2cn(CC(=O)NC3CC(CCC(=O)OC(C)(C)C)C3)nn2)ccccc1Cl 5865,C1(C(N2CCC(CNC(C3C(=C)C3)=O)CC2)=O)OC2CCC1CC2 5866,C1(CC(N2CCC(COC)(CNC(=O)OC(C)(C)C)C2)=O)OCCCC1(C)C 5867,c1(C(n2ccnc2NCC2CNC2)C)cccc(OC(C)(C)C)c1 5868,CC1CN(C(c2cscc2Br)=O)CC1CCNC(=O)CCOC1COC1 5869,n1(CC(=O)NCC2CCCC2C(=O)Nc2cc(O)cc(F)c2)cc([N+](=O)[O-])cn1 5870,CC(C)CCCCC(=O)NCC1CCC1C(N1CCC(n2cncn2)C1)=O 5871,C12(C(=O)NC3C(NC(c4ccc(CO)nc4)=O)COCC3)CCC(CO)(CC1)C2 5872,C=CC(C)CCN=c1[nH]c(=NCC2(C)CC2(F)F)c2cc(Cl)ccc2[nH]1 5873,N1(C(C(COC)C)=O)CCC(CC(C)NC(=O)CN2CCNC(=O)C2)CC1 5874,CCCCC(CN(C(=O)CC=CC(C)(C)C)CC)NC(=O)CCC(=O)NC 5875,C(C(C)C(C)C(=O)NCC(C)CN(C(=O)CC=Cc1ccc(F)cc1)C)OC 5876,C1(O)(CNC(c2ccnc(OC)c2F)=O)CCCN(C(=O)CN2CC=CC2)CC1 5877,N1(C(c2c(CC)ncs2)=O)CC(O)CC1CC(=O)NC1(CN(C)C)CC1 5878,Clc1cccc2c1C(Nc1nnnn1CC1CC(c3ccc(F)cc3)C1)CC2 5879,N1(C(CC=C=C)=O)CCN(C2CCCN(C(=O)C(C(C)C)SCC)C2)C(=O)C1 5880,C1(C(=O)Oc2cccc3c2OCCO3)COc2c(cc(Cl)cc2[N+](=O)[O-])C1 5881,C1(C(=O)NCC(CO)C2CC2)CC(O)CCN1C(=O)CC1CC=CC1 5882,CCCC(O)CC(=O)NC(C)(C)CCCNC(c1cc(-c2ccc(C)s2)[nH]n1)=O 5883,N1(C(=O)OC(C)(C)C)CC2CCC1(C(=O)Nc1ccc(OC(F)F)c(Cl)c1)CC2 5884,c1(C(C(=O)NCC=CCNC(C2CCC(F)C2)=O)(F)F)c(F)cccc1F 5885,N1(CC(=O)N(C(CN(C(C(C)CC2CCCC2)=O)C)C)C)CCCNC1=O 5886,c1(NC(C(Br)=C(C)C)=O)nccc(C(F)(F)F)n1.C12CCCC1CNC2=O 5887,C1(C(=O)NC(C)CNC(=O)C=Cc2cnc(C)s2)(CC)CCC(O)CC1 5888,C1=CCCC(Nc2ncc(-c3ccccn3)s2)CCC1 5889,C(CC(C)(C)CC(=O)N1CCCN(C(=O)Cc2c[nH]c(=N)nc2O)CC1)OC 5890,N1(C(CN(C(C2(CC=C)COC2)=O)C)=O)CCN(C(c2cscc2F)=O)CC1 5891,C1(NC(=O)COc2ccccn2)(CO)CCN(C(c2cn(CC3CC3)nn2)=O)C1 5892,C1(NC(c2nc(COC)sc2)=O)CC2CN(C(=O)COCC3CC3)CC12 5893,N1(C(c2ncc(C)c(C)c2)=O)CCC(C)(C)C(C(=O)NCCc2cccnc2)C1 5894,c1(CNC(c2nc(C)c(C)[nH]2)c2nnnn2C2COC2)cc(Cl)ccc1F 5895,C1(C(C)NCCC2CCCN(C(C)C)C2)CN(C)CCN1C 5896,CCCCCC(O)C(=O)N1CCN(C(c2cnc3occc3c2)=O)C(C(C)C)C1 5897,c1(N2CCC(O)(C(=O)NCC(C)(C)O)C2)ncnn2cccc12 5898,c1(CNC(C2C(NC(c3c(C#N)nc[nH]3)=O)C2)=O)cc2ccccc2o1 5899,c1(C(=O)NC2C3CN(C(C4(SCC)CC4)=O)C2C(O)C3)sc2cccnc2c1Cl 5900,C1(CNC(c2cnoc2)=O)CCN(C(c2cn3ccccc3n2)=O)CC1(F)F 5901,Cc1ccc(C(N2CC(C(F)Cn3cc(C4CCCC4O)nn3)C2)=O)o1 5902,CC1(C)C(CO)CCN1C(=O)CCC1CCN(C(C2CCCOCC2)=O)CC1 5903,N1(C(=O)OC(C)(C)C)C2CCC1CN(C(=O)OCC1CCCN(S(C)(=O)=O)C1)C2 5904,N1(C(C=C(CCC)C)=O)CCC2CN(C(c3cnn(C(C)(C)C)c3)=O)CCC2C1 5905,C1(C(N2C(C(=O)NCC3(OC)CN(C)C3)CCCC2)=O)CCC(C)(C)OC1 5906,C=Cc1cc(C(=O)NCC2CCC(C)CN2C(c2nnc(S)n2C)=O)cc(F)c1 5907,N1(C(C2C(CNC(c3cnn4c3CCC4)=O)OCC2)=O)CCC12CCCOCC2 5908,CCCCC(C(=O)NC1CC(C)N(C(=O)C(CC)C(C)C)C1)NC(N)=O 5909,c1(NC(C2NCCN(S(CCC)(=O)=O)C2)=O)cccc(C(=O)OC)c1C 5910,N1(C(c2ccc(Cl)c(N)c2Cl)=O)CCN(C(=O)C2=NOCC2)C2CCCCC12 5911,c1(N2CCCCC2C2CC2)nc(=NC2CCc3ccccc3C2)[nH]c2c1CSC2 5912,N(C(=NCCc1ncc(C)s1)N1CCCC(CNC(N)=O)C1)C(COC)C 5913,c1(CN(C(c2c(CC)ccs2)=O)C)cnn2c1CN(C(c1c[nH]c(=N)s1)=O)CC2 5914,C(=O)(CCCCC(F)(F)F)NCC(CNC(c1c(C)nn(CCC)c1C)=O)OC 5915,N1(C(CC=CCCCCC)=O)CCCCC1CC(=O)NCC1CCCN1C(C)=O 5916,c1(OC)nscc1C(=O)NC1COCC1NC(C1CC1(C)C)=O 5917,C(=O)(C(CC)CCC)NC(CC=C)CNC(=O)CCC=CC(C)C 5918,c1(C(N(CC(C)NC(c2cnc(CC)o2)=O)CC)=O)ccc(C(F)F)cn1 5919,N1(C(C(=O)NCC)=O)CCN(C(c2sc(C)cc2OC)=O)C(C2CC2)C1 5920,CC(=O)CCCC(=O)NC(C(=O)NCCCOC1CCCC1)C(C)C 5921,C(=O)(C(O)CC(C)C)Nc1ccccc1.CCC(C)(C)OCC(=O)NCC1CC1 5922,N1(C(c2snc(C)c2N)=O)CCC(N=[N+]=[N-])(C(=O)NCC(O)CF)C1 5923,CCC(CC)C(C(=O)NC(C)C(=O)NC(C)(C)CC(C)(C)C)OC 5924,O=[N+]([O-])c1ccc(NCc2cnn(-c3ccccc3)c2)cc1I 5925,N1(C(C2(C)CC(=C)C2)=O)CC2CC2(NC(=O)C(F)=C(C)C)C1 5926,C1(CCNC(C2C(CC)OCC2)=O)CCCN(C(c2cnc(C(C)(C)C)s2)=O)C1 5927,Cc1ccc(O)c(C(=O)NC(C)C(C)(C)NC(C2CCN(C)S2(=O)=O)=O)n1 5928,N1(C(=O)Cc2cn[nH]c2)CC(C2CN(C(=O)CCSc3ccc(F)c(F)c3)C2)C1 5929,C1(C(=O)NCC(n2cc(CN3CC4CC4C3)nn2)C)CCC(=O)C(C)C1(C)C 5930,C1(CC(C)NC(C2CCC(=O)N2C)=O)CCN(C(C2(C)CCCS2)=O)CC1 5931,N1(C(c2cc(C)no2)=O)CCCC(O)(CNC(c2cc(Cl)ncc2N)=O)C1 5932,C1(CN=C(NCC(F)=C(C)C)NC2CCN(C(=O)C3CC3)C2)CCCCC1(F)F 5933,N1(C(C(C(C)C)C)=O)CCC(C)N(C(=O)CCCCOCCO)CC1 5934,S(=O)(=O)(c1ccc(OCC(=O)O)c([N+](=O)[O-])c1)NC1C(C)(CC)CCO1 5935,C12(CNC(=O)Cc3csnn3)CCCC1CCN2C(c1ncccn1)=O 5936,n1(CC(=O)NCC(CNC(c2cc(C)c(C)s2)=O)CO)ncn2nccc2c1=O 5937,C(=O)(CC(C)C(=O)N1CCC(NC(=O)CC2(C)CC2(Cl)Cl)C1C(C)C)OC 5938,c1(C(N)=O)nc(C(N2CCCC2CNC(c2cc(O)cs2)=O)=O)cs1 5939,CC(C#N)CN=C(NCc1cnccc1Cl)NC(c1ccccc1)C 5940,Cc1c(C(=O)NCC2(NC(c3csc(C(F)(F)F)c3)=O)CCC2)cnn1C 5941,C(CC(C(=O)NC(C)C(C)OC)NC(=O)CC1CC1)OC 5942,CC12CCN(CC1)CC2C(=O)NCC1CC(NC(c2cc3ncccc3s2)=O)C1 5943,N(C1c2ccccc2CC1C)C(C1CN(c2c(OC)cccc2)C(=O)C1)=O 5944,c1(C(N2C(CNC(C(C)Cc3ccco3)=O)C=CC2)=O)cc2n(c1)CCC2 5945,C(N=c1nc(N(C)C(C2CCCC2)C)c2c([nH]1)CCOC2)C1(COC)CCC1 5946,S(=O)(=O)(c1cnccc1NCC1(CO)CCOC1)N(C)CCC1N(C)CCC1 5947,c1(C(=O)Nc2c(C)cc(NC(=O)C(C)S(C)(=O)=O)cc2)cc2ncn(C)c2cn1 5948,c1(OC)cc(F)c(F)cc1C(=O)NCCC1(CNC(C23CC4CC2C3C4)=O)CC1 5949,C(=O)(C(Cc1cn[nH]c1)NC(c1cnc(O)o1)=O)N(CCCN(C)C)CC 5950,C12(C3CCN(CC3)C1)CC2.C=CC(CC)CC(=O)NCCCC(=O)OC 5951,C1(NC(C(C)(N(C(=O)C(=O)C(C)(C)C)C)C2CC2)=O)CCCOC12CCC2 5952,c1(CC)ccc(Br)cc1C(=O)NC(C)CCN(C)C(C1C(C)(C)C1(C)C)=O 5953,CN1CC(NC(=O)NCC23CC(C2)C(C(F)(F)F)O3)Cc2ccccc21 5954,c1(C(=O)Nc2ccncc2)nc2n(c1Cl)CCN(C(c1cc(Cl)ccc1Br)=O)C2 5955,C1(C)(NC(CC2CCN(C(C(C)OCC)=O)C2)=O)CCC(C)(C)C1 5956,c1(-n2c(CC3SC(=N)NC3=O)nc(COC(C)C)n2)ccc(Cl)c(F)c1 5957,C1(NC(C(C)CO)=O)CN(C(c2cc3n(n2)CCCO3)=O)CC12CCC2 5958,N#Cc1cncc(NC2(c3nnnn3CCCF)CCN(C(=O)N(C)C)CC2)c1 5959,c1(CC(C(=O)NC(C)CCCNC(C2CC2(C)C(C)C)=O)=O)ccc(F)cc1 5960,Cc1ncc(Cl)cc1C(N1CC(N(C(=O)CC2CCCCC2(C)C)C)C1)=O 5961,N1(C(CCc2n(C)ncc2)=O)CCC(C(N2CC(O)(C(F)F)C2)=O)C12CC2 5962,S(=O)(=O)(c1cccc(=NCCCSC(C)(C)C)[nH]1)N1CCC(OCC(C)C)C1 5963,c1(CC)cnoc1C(=O)NCCN(CCC(=O)NC1CC1)C 5964,c1(CC(N2CCC(NC(C3(CCC)CC3)=O)C2C(C)C)=O)ccc(S(N)(=O)=O)s1 5965,c1(C(N2CCC(C(C)(C)NC(CCOC(C)=O)=O)C2)=O)cn(C(C)C)nc1C 5966,c1(OC)cc(C(N2CCC(C(=O)Nc3cccnc3C(F)(F)F)C2)=O)cc(Br)c1 5967,c1(C(=O)NCC2CCCN(C(C3C(C#C)C3)=O)C2)cc2sc(Cl)cc2s1 5968,N1(C(CCC)=O)CCC(N(C2CCC2)C(C2CCCN2C(=O)OC)=O)C1 5969,CC(C(C)C(=O)NCc1ccc(CNC(=O)CCS(C)(=O)=O)cn1)C(C)(C)C 5970,c1(SCC)cccc(C(=O)NCCCC(C)NC(=O)CCC2CC2(C)C)c1 5971,c1(NC(CCCC)CC)ncnc(NC(c2cc(C)oc2C)C)c1C 5972,O(NC(=O)C(CNC(C1CCCSC1C)=O)N(C)C)CCCOCC 5973,C1(n2ccc(C)n2)CCN(C(=NCc2ccco2)NCC2C(C)C2C)CC1 5974,c1(-n2c(C3C(C)C3C)nc(CC(C)OC)n2)ccc(F)c(Cl)c1 5975,CC1CCN(C(=O)CC(C2CCC2)C2CCC2)C1CNC(=O)CC1OCCCO1 5976,C1(C)(C(N2CCC(O)(CN(C(=O)C3=CCOC3)C)CC2)=O)CC(C(C)(C)C)=NO1 5977,C12(C(N(C)CC3(CC(C)C)CC3)=O)CC(CNC(c3nnc(S)n3C)=O)(CO1)C2 5978,c1(C(=O)NC2CC(NC(=O)CCc3nccs3)C2)ccc(CO)nc1 5979,c1(OCCOC)ccc(CC(N)=O)cc1.C1(COC(C)(C)C)CCOC(=O)N1 5980,c1(CC(C)C)ccc(C(C)C(=O)NCC2CN(C(C3CCCOC3C)=O)C2)cc1 5981,c1(C(=O)NC2CC(NC(=O)Cn3ncccc3=O)C2)cccc2c1C(=O)NC2 5982,C1(CC)CN(C(=O)C(c2ccccc2)C)CCC1N=c1[nH]c2ccc(Cl)cc2s1 5983,S(=O)(=O)(c1cnn(C)c1)N(C)CC1CCC(=O)NC1.C12CCN(C1)C(=O)CN2C 5984,CC1CC(C(=O)NCC(C)(C)NC(=O)CCc2ccc(F)cc2)=NO1 5985,N1(C(c2c(C)cc(CO)o2)=O)CC(C2(NC(=O)CC(C)CN(C)C)CC2)C1 5986,CC#CCCCC(=O)NCC1CN(C(c2c(Br)ncn2C)=O)CCCO1 5987,c1(C(n2cc(C3CCN(C(C4COCCO4)=O)C3)nn2)CC)ccccc1F 5988,C1(C(=O)NC2C=CCN(C(c3nnc(C)s3)=O)C2)Cc2ccccc2C1 5989,C(=O)(C(F)(F)CCn1cccn1)NCC1(NC(C2C(C)(C(F)F)C2)=O)CCC1 5990,c1(-n2cc(C(N(C(CC)=O)C)C)nn2)c(C)cccc1[N+](=O)[O-] 5991,C(=O)(C(CC(F)F)N(C)C(c1ccc(C)nc1)=O)NC1CCCC(OC)C1 5992,C1(OCC(=O)NC2CN(C(C3(C(F)(F)F)CCOCC3)=O)C2)(CO)CCOCC1 5993,c1(C(=O)NC(C2OCCN(C(C(=C)F)=O)C2)C)ccc(S(=O)(=O)N(C)C)cc1 5994,CC(C(=O)NCCOCCCNC(C1CC(=O)NC(=O)N1)=O)C(C)S(C)(=O)=O 5995,n1(CC)cccc1C(=O)NCC(CCNC(c1ccc(CO)o1)=O)OC 5996,C(=O)(C1=CS(=O)CCC1)N(CCCNC(C(CC=C)C)=O)Cc1cccnc1 5997,c1(C(N2CC(NC(CC(CC)CC)=O)C(C)C2)=O)ccc2c(c1)N(C)CC2 5998,C(C(=O)N1Cc2ccccc2CO1)C1CC(NC(CCC=C(C)C)=O)C1 5999,Cc1ccc(N(C(=O)CC2CCCN2C(C2CC3CC3C2)=O)C)c(C)c1 6000,c1(CN2CC(C#N)C(NC(c3ccc(S)cc3)=O)C2)cc(Br)cc(F)c1F 6001,c1(C(=O)NC2(CC)CN(C(=O)CN3CCCCC3=O)C2)ncncc1C 6002,N1(C(C(CO)OC)=O)CCC(C(=O)NCC2CCN(C3CC3)C2)CC1(C)C 6003,N1(C(C(C)NC(=O)OC)=O)CCOCC1C(N1CC(F)(F)C1C1CC1)=O 6004,c1(CC(=O)N(CCOC)C)c[nH]c2ccc(-c3cc(C)c(OC)c(C)c3)cc12 6005,C(=O)(C1=NN(C(C)C)C(=O)CC1)NCCCC(C)NC(C=C(COC)C)=O 6006,C(=O)(C1CCCn2nccc21)N1CC2N(C(c3cc(C)cc(Cl)c3)=O)C(CC2)C1 6007,C(N=c1[nH]c(N(C)CCC2CCC2)nc2ccc(Cl)cc12)c1n(CC)cnc1 6008,Cc1cc(CNC(C2CC(C)N2C(=O)CCC2(C)CC2)=O)ccc1F 6009,CC(C)CC(C(=O)O)NC(C1CCCN(C(c2ccnn2C)=O)C1)=O 6010,c1(CNC(C=CC(=O)N(C)C)=O)nc(CNC(=O)CN(C)C2CC2)cc(O)n1 6011,c1(NC(=O)NCc2csc(CO)n2)cc2c(nc1O)CCC2 6012,c1(C(=O)NC2C(CNC(C(C)SC)=O)C2)ccc(-n2cccn2)nc1 6013,N1(C(C(COC)OC)=O)C2CCC1CC(NC(c1ccccc1SC(C)C)=O)C2 6014,C1(C(=O)NCCC(C)O)COCCN(C(=O)CCc2cccnc2)C1 6015,CCC(O)C(C)(C)C(=O)NCCCN(C(=O)COc1ccc(CO)cc1)CCO 6016,c1(SC)nc(C)c(Br)c(=NCc2cc(C(F)(F)F)cc(C(C)(C)C)c2C(C)(C)C)[nH]1 6017,C1(CC(=O)NCc2cn[nH]c2)CCN(C(C2CCO2)=O)CC1 6018,N1(C(CCSCCC)=O)CC(NC(c2c(C)csc2Cl)=O)CC1(C)CC 6019,C(=O)(CCCC(=O)N1CCC2CCC12CNC(c1ncc(F)cc1F)=O)N(C)C 6020,C1(C(=O)NCCCCNC(=O)C=Cc2cccnc2)CCC(=O)N2CCCC12 6021,N1(C(C2CC23CCC3)=O)CC2CCC(C1)N2C(=O)C(O)CC1CCCCC1 6022,CCC(C)(O)CNC(=O)CCCC1(NC(=O)COCCF)CCC1 6023,Cc1nc(C(N2CC3CC2CN3C(=O)CSCCC#N)=O)c2ccccn12 6024,C1(C)(C(=O)NC2C(NC(C(c3ccccc3)OCC)=O)CCC2)CC=C(C)CC1 6025,c1(N(C)CC2CC2(F)F)cccc(S(=O)(=O)N2CCSC(c3ccccc3)C2)n1 6026,CCCCC(CN=c1[nH]nc(Cc2ccccc2)s1)NC(=O)CSCCC(C)C 6027,C(CCCCC(=O)N(C)CC1(O)CCCN(C(=O)CC2CC(F)C2)C1)OCC 6028,C1(N(C(c2cncc(C)n2)=O)C)CCCN(C(c2cc(Br)nn2C)=O)CC1 6029,c1(C(=O)NC(C(=O)NC(C=C)CO)c2ccco2)cnccn1 6030,S(=O)(=O)(c1c(F)cc(F)cc1F)Nc1scc(C(=O)Nc2cccc(Br)c2F)n1 6031,CCCCC(C(=O)NCc1cc(C2CC2)no1)NC(C1OCCC1(C)C)=O 6032,n1(CCCNC(C(=O)Nc2cccc(C(=O)OC)c2Cl)=O)c(C)cc(C)nc1=O 6033,c1(C(=O)NC2CN(C(C3C(C)CCC3)=O)CC2F)cn2ccc(Br)cc2n1 6034,C1(O)(CN(C(C(C)SC(C)C)=O)C)CCN(C(c2n[nH]c(C3CC3)c2Cl)=O)C1 6035,C=CCC(CC)C(=O)N1CCN(C(=O)CN(C(=O)COC)C)CC1C(C)C 6036,C1(C(=O)NC(C)Cc2nc(-c3ccccc3)no2)CC(O)C(O)C1 6037,N1(CC(C)C)CCC(C(N2CCCC(CN(C)C(C3(CO)CC3)=O)C2)=O)CC1 6038,Cc1cc(C(=O)NC2CC(C)(NC(C3CCCN(C)C3)=O)C2)c2sc(=N)[nH]c2n1 6039,N1(C(C(C)OCC#C)=O)Cc2cccc(CNC(=O)C(CC)CCCCC)c2C1 6040,Cc1nc(NC(C2(C)CCN(Cc3ccncc3O)C2)=O)ccc1Br 6041,c1(N2CCC(CNC(=O)CCOCC3CCCO3)C2)ncc2ccccc2n1 6042,c1(C(=O)NC2CCN(C(C(C3CCC3)OC)=O)C2C(C)C)coc(S(C)(=O)=O)c1 6043,C1(C(=O)NCC(CNC(c2n(C)cnn2)=O)O)CCn2ncnc2C1 6044,N1(C(CC2(C=C)CC2)=O)CCCC2(NC(C3CCC(C(N)=O)CC3)=O)CC2C1 6045,c1(C(=O)NC2CN(C(c3coc(C4CC4)n3)=O)C3CC23)cc2scnc2[nH]1 6046,C1(C(=O)NC2CC(NC(=O)CCC3CCCCC3)C2)CCCN(C(=O)C2CC2)C1 6047,c1(CC(=O)NC2C(NC(C(C(C)C)NC(N)=O)=O)COC2)nn(C)cc1[N+](=O)[O-] 6048,CCCCC(CNC(=O)CC(O)Cc1ccccc1)NC(C1(F)CC=CC1)=O 6049,C(N=c1nc(N2CC3CCN(C)CC3C2)c2[nH]ccc2[nH]1)c1c(OC)cncc1 6050,c1(Cn2cc(C(c3nnnn3CC(F)F)NC(CC)C)nn2)c(C)cccc1Br 6051,N1(C(C=Cc2c(C)nccc2)=O)CCCC2(CCCCC2NC(=O)CNC=O)C1 6052,Nc1c(F)c(F)cc(C(N2CCN(C(C3CC(O)C3)=O)C3CCC23)=O)c1Cl 6053,CC(CCC(=O)Nc1cn(C)nc1Cl)NC(c1ccncc1Cl)=O 6054,c1(OCC)ccc(C)nc1C(=O)NCC1CC1NC(c1cc([N+](=O)[O-])c[nH]1)=O 6055,c1(C(N(C2CCCN(C(C3CCCN3C)=O)CC2)C)=O)cc2ccc(F)cc2s1 6056,Cc1cc(F)c(C(=O)NC2CC(CCNC(C3CCOC3C)=O)C2)cc1F 6057,C1(C2CC2)(C(=O)NCCCCNC(=O)C=CCN2CCOCC2)CCC1 6058,C(=O)(C1SCCc2sccc21)N1CCC2(CC(NC(=O)CC=C(Cl)Cl)C2)C1 6059,c1(C(=O)NC2C(NC(=O)OC(C)(C)C)CCC2)ncc(Br)cc1O 6060,C1(C(N2CC(O)(CCNC(c3cn(CC)nc3)=O)C2)=O)CCc2nnn(C)c2C1 6061,O=C(C(F)C1=CCCCC1)NCC1CC2CCC1N2C(=O)Cc1ccc(Cl)cc1 6062,c1(OC)ncc(Cl)c(C(N2CC3(NC(=O)C(C(C)C)SC)CC2C3)=O)c1Cl 6063,c1(OC)nccc(C(=O)NC(C)(C)C(C)NC(=O)C2=CCCC2C)c1Br 6064,Cc1nc(CO)ncc1C(N1CCC(NC(C2C=CCCC2)=O)C1(C)C)=O 6065,c1(C(=O)NCC(C2CCOC2)NC(CCC(N)=O)=O)cnc2ccccn2c1=O 6066,C(=O)(C1=CC2(CCOCC2)C1)NCC1CC(C)N(C(=O)C=C2CCCCC2)C1 6067,S(=O)(=O)(c1cccnc1NC1CCCC1c1ccccc1)N(C1(C)CCCC1)C 6068,C1(C)(CNC(C(C2CN(C(c3cnc(C)s3)=O)C2)O)=O)CCN(C)C1 6069,C1(C(=O)NC2CC(NC(c3ccn(C(C)C)n3)=O)C2)CCN(CCO)C(=O)C1 6070,C=CCCCCCCCC(=O)N1CC2CC1CC2NC(=O)C1CC1 6071,N1(C(C(C)CC2CCCO2)=O)C2CCC1CN(C(=O)CN1CC(C)(OC)C1)C2 6072,c1(C(=O)NC(C(C)NC(Cc2c(C)n[nH]c2C)=O)(C)C)cnn2c1OCC(C)C2 6073,c1(CC2(C(=O)NC3CC(O)(CNC(C4CCCO4)=O)C3)CC2)cccc(F)c1 6074,N1(C(CCc2cn(C)nc2)=O)CCC(NC(=O)CSc2cn[nH]c2)C1C1CC1 6075,C(=O)(C(CNC(=O)C1=C(C)OCC1)C(C)C)NCc1cnc(CC)s1 6076,C1(CNC(COC)=O)CC2CC1CN2C(c1ccc(-c2ccsc2)cc1)=O 6077,Cc1nn(CC(N2CC(NC(c3ncc(F)cn3)=O)C(C)C2)=O)cc1Br 6078,C1(NC(C(n2ncc(C)c2)C)=O)CCCCC1NC(=O)C=Cc1ccoc1 6079,C(=O)(C(F)(CNC(C1CC(C(=O)OC)C1)=O)C(C)C)N(c1cccc(CC)c1)C 6080,N1(C(C=C(CC)C)=O)CCN(C(=O)COC2CC(F)(F)C2)CC1CC 6081,N1(CC)CCOC(C(=O)N(C(=O)C(C)Oc2cccc(CSC)c2)C)C1 6082,C(=O)(C(C)(C)C(=O)Nc1ccc(F)c(F)c1)N1C(CNC(CCC=C=C)=O)CC1 6083,c1(C(CC)C)ccc(C(=O)NCC(C(C)C)NC(C2(O)CC2)=O)c(O)n1 6084,c1(NCC2(NC(=O)OC(C)(C)C)CC2)n[nH]c(=N)[nH]1 6085,C1(C2CC2)(NC(CN(CCC)C(C2CC2C(F)(F)F)=O)=O)CCCC1 6086,c1(NC(c2ccc(OC(F)(F)Cl)cc2)=O)cccc(-c2nc(O)n[nH]2)c1 6087,c1(COC)cc(N(CC(C)CNC(C2CCCOCC2)=O)C)nc(SC)n1 6088,CCCCC(CN1CCCC(C(N2CCCC(CO)C2)=O)CC1)CC 6089,CP(C)(=O)C1CCCN(C(=O)NCC(c2ccccc2)C2CC2)C1 6090,N1(C(C(CC2CC2)NC(C2CN(C3CCC3)C2)=O)=O)CC2(CCC2)C1 6091,CS(C)(=O)=Nc1nc(C(=O)NC2CCN(C(=O)C=Cc3cnc[nH]3)C23CC3)cs1 6092,C1(NC(CCC(C)OC)=O)CC2CCC(C1C)N2C(=O)C1=CCCCO1 6093,C1(C(=O)NCCCN(C(C2CS(=O)(=O)C2)=O)CC)CCC1(F)F 6094,CC1=CCSC1C(=O)NC(C1CCN(C(=O)CC2CCCC2O)C1)(C)C 6095,C1(CC=C)(NC(c2nc(Cl)c(CC)[nH]2)=O)CCN(C(C2(CN(C)C)CC2)=O)C1 6096,C1(C(N2CCC(Cn3cc(C(CCC)=O)nn3)C2)=O)CS(=O)(=O)C12CCOCC2 6097,N(C1c2ccccc2CC1NC(=O)C(O)C1CC1(Cl)Cl)C(C(C)(C)N1CCC1)=O 6098,CCCC(CC)C(=O)NCCC1(NC(=O)C2=NNC(=O)C2)CCCC1 6099,C1(NC(C(CC)CC2CCCC2)=O)CC2CN(C(c3ccccc3CO)=O)CC2C1 6100,N1(C(C(C)N(C(C2CC(CCC)C2)=O)CCC)=O)CCOC2C(O)CC12 6101,C1(NC(C(CC=C)C)=O)CC(OC)CN(C(c2cc(C)n(CC)n2)=O)C1 6102,C=CCCC(C(=O)N1CCCC1COC)NC(=O)C(CN(C)C)N(C)C 6103,C1(NC(c2c(OC)csc2)=O)CC2CN(C(c3ccc(CO)s3)=O)CC2C1 6104,N1(C(COCC=C)=O)CCC(CNC(c2cccc(C)c2)=O)C12CCC2 6105,N1(C(=O)C=Cc2cocn2)CCCC12CCN(C(=O)C(F)(F)CC1CC1)CC2 6106,C1(CNC(Cc2c(C)con2)=O)(CNC(c2cc(C)n(CO)n2)=O)CC12CCC2 6107,S(=O)(=O)(CC(=O)NC(CNC(c1ccnnc1NC1CC1)=O)C1CC1)NCC(N)=O 6108,C1(CNC(C2CCCCCC2)=O)C2CCCC1N(c1cc(Cl)c(O)nn1)C2 6109,C1(CNC(C(COC)OC)=O)CCC2(CN(C(=O)Cc3cncc(O)c3)C2)O1 6110,N1(C(c2c(C)n[nH]c2)=O)CC=CC(NC(c2ccc(C3CCC3)nc2)=O)C1 6111,Cc1ccnc(C(N2CCC(N(C(=O)CN3CCCCCC3)CCO)C2)=O)c1N 6112,Cc1cncc(C)c1C(N1CCCCC1CNC(c1ccc(C#N)cn1)=O)=O 6113,C(CCCCCNC(=O)CC1CC(NC(=O)Cn2ncn(C)c2=O)C1)OC 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6204,C1(C)(CNC(c2c(C)ncs2)=O)CCCN(C(=O)Cc2csc(NC=O)n2)C1 6205,Cc1cncc2cc(C(N3CCCOC(CNC(=O)Cc4csnn4)C3)=O)sc12 6206,N1(C(c2snc(C)c2N)=O)CCCN(CCNC(C2CN(C)C2)=O)CC1 6207,O=C1CCC(C(=O)N2CCC(NC(c3cc(C(F)(F)F)cc(Cl)c3)=O)C2)=NN1 6208,C1(NC(c2nc(C)sc2)=O)COC2(CNC(=O)CCOC3CCCOC3)CC1C2 6209,N1(C(C(F)=C(C)C)=O)CCC2CN(C(c3cc(Br)n(C)n3)=O)CC2C1 6210,C1(NC(C2CC3CC2C2CC32)=O)CCCCN(C(c2cc3occc3[nH]2)=O)C1 6211,N1(C(c2c(N)cccn2)=O)CCC2(CCOC2)C(CNC(c2csc(Cl)n2)=O)C1 6212,C12(CNC(C(COC)O)=O)CCCCC1N(C(c1cc(OC)nn1C)=O)CC2 6213,C1(C(N2CC(CC(C)NC(C(C)C)=O)C2)=O)(N(C)C)CCCCC1 6214,C(=O)(C(CC(C)(C)C)NC(=O)C(C1(O)CCCC1)F)N1CC(SCC)C1 6215,C(CCCCNC(=O)COCC(C)(C)C)N(C(CCC1CC(C)C1)=O)C 6216,c1(C(=O)NC2CCC(NC(Cc3ccn(CC)n3)=O)C2)ccc(C)c(C)c1N 6217,c1(CNC(c2c(C(C)(C)NC(=O)C=CCO)noc2)=O)ccccc1F 6218,C1(COC)CC(O)CN1C(=O)C(C)N(C(=O)Cn1ncccc1=O)C 6219,N1(C(c2ccn(CCNC(c3c(C)cc[nH]3)=O)c2)=O)CCC(CO)(CO)C1 6220,C=CCCC(=O)NC(CNC(C1CN(C2CCOC2)C1)=O)C1CCC1 6221,CCCCCCC(C)C(=O)N(C1CN(C(c2cc(C#N)cn2C)=O)CC1(C)C)C 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6240,S(=O)(=O)(c1cnc(NCc2csc(C(C)(C)C)n2)cc1C)NC(COC)CCO 6241,C(CC(=O)NCCCCCSC)(C(F)(F)F)NC(c1c(CC)cc[nH]1)=O 6242,CCC(C)(COC)C(=O)N1CC=CC(NC(=O)C(C)(C)C(F)F)C1 6243,C1(C(=O)NCC(C)(CO)NC(Cc2c(Cl)cn(C)n2)=O)CCCCC(F)(F)C1 6244,C(=O)(C(O)CC1CCOCC1)NCCN(CCC)C(C1(CO)CCCO1)=O 6245,Cn1nncc1C(=O)NCC1(NC(=O)Cn2ccnn2)CCOC1 6246,c1(C(=O)NCCN(CCC)C(C)C)cc(Cl)ncc1F 6247,c1(C(=O)NCC(C2CC2)NC(c2cccnc2S)=O)cc2ccsc2s1 6248,CC1(CC(=O)NCC2CC2NC(c2cccc(OCCF)c2)=O)CCS(=O)(=O)N1 6249,c1(C(N(CC(C)(C)NC(C(CC)n2ccnc2)=O)C)=O)cnc2ccoc2c1 6250,C=CCCCCC(=O)NCC(O)CCNC(=O)C(CCCC)NC(N)=O 6251,N1(C(CSCC)=O)CCCC2C1CCN2C(c1c[nH]c(Br)c1)=O 6252,c1(C(N2CCC(CNC(CSc3cn(C)nc3)=O)C2)=O)cccc2oncc12 6253,CC(CCF)N=c1nc(N(C)CCN(c2cccs2)C)c2cc(OC)ccc2[nH]1 6254,C=C(C)CCC(=O)N(C1C2CN(CC(F)(F)F)CC12)C(C1(C(=O)OC)CC2CC2C1)=O 6255,Cc1cc(OC(F)F)ccc1F.C12CN(CC1C)C(=O)COCC(=O)N2 6256,c1(C(=O)OC)c(C)[nH]c(C(N2CC(NC(=O)C(C)CSc3ccccc3)C2)=O)c1C 6257,C(=O)(CC(CC)CC(C)C)NCCC(=C)CNC(c1ccc(F)cc1)=O 6258,O=S(=O)(c1ccc(Cl)c(F)c1F)N1CCCCCC1CC(c1cccs1)O 6259,c1(C(=O)NC(C)C(C)NC(c2ncccn2)=O)ccc(N2CCCC2=O)cc1 6260,CCC(CC)C(C)C(=O)N1CCC(C(C)CNC(c2nc(C)ncc2Cl)=O)CC1 6261,C1(C(N2CCC(NC(C3CC(F)(F)C34CCC4)=O)C2)=O)Cc2ccccc2C1 6262,Cc1ccnc(C=CCNC(C2CCN(c3ccccc3)C2)=O)c1 6263,N1(CC)CCCCCC1CCO.N12CC3C(C3C1)C2=O.C1(C)C(=O)NCCS1 6264,c1(NCC)ccc(Cl)cc1C(=O)NCC(F)CNC(C1CC2CC1CO2)=O 6265,N1(C(C2CC=CCC2)C(=O)N(c2c(C)cccc2)C2CC2)CCS(=O)C(C)(C)C1 6266,C(=O)(CC=C(Cl)Cl)NCCC(C)N(C)C(c1ccccc1OCC1CCCO1)=O 6267,CSC1=C(C(=O)NCC(C2CCC2)NC(=O)CC2=NN(C)C(=O)C2)CCCC1 6268,N1(C(CC2CCN(OC)CC2)=O)CCCC(O)(CNC(c2ccncc2)=O)CC1 6269,N1(C(C(C)CN(C)C)=O)CC2CCC1C(CNC(C1(C3CC3)CCCO1)=O)C2 6270,c1(C(N2C(C)C(C)(C)CCC2)C(=O)NC2CC2)cc2ccc(OC(F)F)cc2o1 6271,C(=O)(C(C(F)(F)F)C(F)(F)F)N1CCOCC(NC(c2ccn(CC)n2)=O)C1 6272,c1(SC)ccc(S(=O)(=O)NC(C2C(Cl)(Cl)C23CC3)=O)c(C)c1 6273,c1(C(=O)NCCCOCC=C)cc(CNC(=O)CCCF)ccn1 6274,N1(C(CCCC)=O)CC2CN(Cc3cccc(CC)c3)CC2C1 6275,CCC(C(=O)NC(C)(CNC(C1CCOC1=O)=O)C1CC1)OC 6276,C(C(C(=O)N1CCC1NC(=O)C(Cc1ccccc1)SC)N(C)C)OC 6277,c1(C(=O)NCC2CCCN2C(C2(O)CCOCC2)=O)cccc(Br)c1F 6278,c1(CC)cc(C(=O)NC(C2CCCC2)CNC(C2CC3CCC3C2)=O)cc(O)n1 6279,C12(C(=O)OC)CC(C(=O)NCC(CNC(=O)CN3CCC3C)CO)(C1)OC2(C)C 6280,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CCCC(N(C)C(c2nn(C)cc2Cl)=O)C1 6281,c1(N(C(=O)COC(=O)CC(F)(F)F)CC)cc(Cl)ccc1O 6282,N1(C(C2C(CC)C2)=O)CCN(CC(N2CCC(C3(C)N=N3)C2)=O)CC1 6283,Fc1ccc(I)cc1C(NC1(CCC(F)(F)F)CC1)NC 6284,C(=O)(C1=COCC1)NCC1(F)CC(CNC(C2(CC=C)CCC2)=O)C1 6285,CCCC(C(O)C(=O)N(OC)C(C)CC)NC(c1nccs1)=O 6286,c1(NC)cnc(C(=O)NC(C)(C)CNC(=O)C=C2CCC(C)C2)cn1 6287,Cc1ncccc1C(=O)N(C1CC(NC(c2cc(C(C)(F)F)n[nH]2)=O)C1)C 6288,c1(CC)ccc(S(=O)(=O)N2CCC(C)(C(=O)Nc3c(C)ccc(I)c3C)C2)cc1 6289,CC(CN(C)C)C(=O)NCc1occc1C(=O)NCC1(C)CCCO1 6290,C1(NC(c2cc(CC)no2)=O)CCN(C(C2CC3CC2C3)=O)C1(C)C 6291,C1(C(=O)NCc2cccc(NC(CNC(=O)NC)=O)c2)CCCCN(C)C1=O 6292,C1(NC(c2c(C(C)C)ocn2)=O)CC2CC(NC(c3scnc3C(C)C)=O)CC12 6293,c1(OCC(N2CC(CNC(C3CCCN(C(N)=O)C3)=O)C2)=O)ccc(Cl)cc1Cl 6294,c1(C(N2CCC(CC(=O)NCC(c3ccco3)O)C2)=O)ccc(F)c(F)c1 6295,CCC(CC)(CC(=O)OC)C(=O)NC1CCCN(C(=O)CC(=O)NC2CC2)CC1 6296,c1(C(N2C(CNC(c3ccc(O)cn3)=O)CCC2)=O)cn2cccc(Br)c2n1 6297,c1(CCC(=O)NCC(C)(C(C)C)NC(CCC(=C)C)=O)nnc(S)nc1O 6298,CC1(NC(=O)CCc2ccc(F)cc2)CCN(C(=O)C(F)C2CC2)CC1 6299,c1(C(N2CCN(C(C3(CO)CCCO3)=O)CC2)=O)ncc(F)cc1F 6300,Cc1cc(Cl)c(C(=O)NC2CCC(CNC(C3CNC(=O)N3C)=O)C2)cc1N 6301,C(=O)(C(C)C(=O)N1CCC(C)(C(=O)NCC2(CF)CC(F)(F)C2)C1)OC 6302,N1(C(CC(C)c2ccncc2)=O)CCC2(CC1)CC2CNC(=O)Cn1ccnn1 6303,C1(c2nnnn2CCC2CC2)(NC(C(=O)NCC)(C)C)CCN(C=O)CC1 6304,N1(C(CC2(OC)CC2)=O)CC2CC1C2NC(c1ccnc(-n2ccnc2C)c1)=O 6305,CC(F)(F)CCC(=O)NC1CC2(C1)CC2NC(C1(O)CN(C(=O)OC(C)(C)C)C1)=O 6306,C1(NC(CC(CC)SC)=O)C2CC3C1C3C2C(=O)NC(c1ccccc1)C 6307,C(=O)(CCS(C)(=O)=O)NCC1(CC(=O)NCCC=C=C)CC1 6308,N1(C(C(C)=C2CCCC2)=O)CCN(C(=O)C(=O)NC2CC2)CC1c1cnn(C)c1 6309,c1(SCC(=O)NC(CC)CNC(c2cnn(C(C)(C)C)c2)=O)cccc(Br)c1 6310,Cc1cc(N)ccc1C(N1CCN(C(=O)Cc2ccn(C)n2)CC1C1CCC1)=O 6311,Cc1cccc(OCC(=O)NC(CNC(=O)C(N2CCOCC2)C)CO)c1F 6312,C1(CC=C)(NC(c2csc(C(C)(C)C)n2)=O)CCN(C(=O)C(C2CC2)OC)CC1 6313,N1(C(C(C)C)=O)CCC2(CC1)CC2CNC(C1CCn2cncc2C1)=O 6314,C1(CN)CC2(CC(NC(=O)NC3CCCC(C(N)=O)C3)CCS2(=O)=O)C1 6315,c1(C(=O)NC(c2ccc(C)cc2)C2C3CNCC23)cnc2n1CCS2 6316,C1(OCC)(COC(=O)C=Cc2cn(C)cn2)CCSCC1 6317,N1(C(c2n(C)nc(C3CC3)c2)=O)CC2CC(C1)C2N=c1[nH]nc(C(N)=O)s1 6318,Cc1cncc(OCC(=O)NCC2(C)CCN(C(=O)CC3(O)CCC3)C2)n1 6319,C1(CNC(Cc2ccc(C)cc2)=O)CN(C(c2ncnc(O)c2F)=O)C(C)(C)C1 6320,C(=O)(C(C)(C1CCC1)NC(C1CC1(C)C(F)F)=O)N(CCNC(C(C)C)=O)C 6321,C1(N(C(c2n(CC)ccc2)=O)C)CN(C(c2ncoc2Br)=O)CCC1C 6322,CC1CCN(C(=O)CC2CCC(=O)N2)C(CNC(C2CC(OC(C)(C)C)C2)=O)C1 6323,c1(CNC(C2C(C)(C)CO2)=O)nc(CNC(C2(CCO)CC2)=O)cc(O)n1 6324,C1(N(C(c2cc(CC)no2)=O)CCO)CCCN(C(c2n[nH]c(C)c2F)=O)C1 6325,C(CCN(C(=O)COC1(C)CCC1)C)(C(C)C)NC(CC1(OC)CCCC1)=O 6326,N1(C(C(CCC)C)=O)CC2CCC1C1CN(C(=O)CC3CCS(=O)(=O)C3)CC21 6327,Cc1ccc(C(N2CCC(CN(C)C(C3CC(=O)NC3(C)C)=O)C2)=O)cc1CO 6328,CCCCC(F)C(=O)NC1CCCCC1C(=O)NCc1cc(C)nn1C 6329,C1(OC)CC(F)CN(C(C2CCC(C)N2C(=O)CCn2cnccc2=O)=O)C1 6330,C1(N(C)C)(C(=O)NCCc2csnc2Cl)CCCC1 6331,c1(NC2(CNC(C3C(C)CCCC3)=O)COC2)cc(C2CC2)nc(SC)n1 6332,C(=O)(CC(C)(O)C(F)(F)F)N1C2CC(N(C)C(C3CC(O)C3)=O)CC1CC2 6333,C(C(C)(C)CC(=O)N(CC(C)(C)CNC(c1ccn(C2CCC2)n1)=O)C)N(C)C 6334,C1(CC=C)(NC(=O)CC2CCCCC2O)CCN(C(=O)C(O)CCSC)C1 6335,Cc1c(C(=O)NCC2C3CN(C(c4nccn4C)=O)CC23)ccn1C 6336,c1(C(=O)NC2C(NC(c3c(COC)cc[nH]3)=O)CC2)ccc2c(c1)NC(=O)CS2 6337,N1(C(C(C)NC(=O)NC)=O)CCC(C)(CC(=O)NCC(C)CO)C1 6338,N1(C(C=CCC)=O)CC(O)C(O)C1CNC(=O)CCc1cccs1 6339,CC1(C)COc2cc(Br)ccc2C1NC(C1CCN(c2ccc(Cl)cc2)CC1)=O 6340,c1(CCNC(C(C)=CC2CC2)=O)ncnc(N2CCOCC2)c1[N+](=O)[O-] 6341,c1(OC)ccc(OCCCC(=O)N(C(C)(C)C)CCN)cc1.C12CCCC1C(=O)N2 6342,N1(C(C(F)=CC)=O)CC(NC(=O)Cn2cnc(Br)n2)CC(O)C1 6343,C(=O)(C(C)(C)CCC#N)NC(C)CN(C)C(c1cn(-c2ncccn2)cn1)=O 6344,N1(C(C(C)C2CCC2)=O)CCCC(CO)(NC(=O)C(C)Cc2ccc(F)cc2)C1 6345,CCCCCC(F)C(=O)NCC1CN(C(=O)COC2CCCCC2)CC12CCC2 6346,N1(C(C2N(CC)CC2)=O)CCN(C(C2CCN(C)CC2)=O)CC1CC(F)F 6347,C1(O)(CNC(Cc2cc(C)[nH]n2)=O)CCN(C(C2CC2c2ccccc2)=O)CC1 6348,C1(NC(CC(C)(C)OC)=O)CC2CCC(C1)N2C(=O)Cc1ccc(C(C)C)cc1 6349,C1(C(N2CCC(CCCC)C2)=O)CCCN(CC(c2cncnc2C)=O)C1 6350,c1(C(=O)NCCN(C(c2c(OC)n[nH]c2)=O)CC2CC2)cn2cc(C)sc2n1 6351,c1(C(=O)NCC(C)NC(=O)CCc2ccccn2)cc(F)c(F)c(N)c1Cl 6352,N1(C(c2c(COC)noc2)=O)CC2(CCN(C(c3ccc(CN(C)C)[nH]3)=O)C2)C1 6353,N1(C(=O)Nc2ccc(OC(C)C)cn2)CC2(CC2)c2ccc(Br)cc21 6354,c1(NC23C(CN(C(c4scc(OC)c4)=O)C2)CCC3)nc2ccc(F)cc2o1 6355,C1(NC(=O)CN(C(=O)CCC2OCCO2)C2CCC2)CCC2CC12 6356,C1(NC(C(C2CCCCC2)OC)=O)CCNC(=O)CC1 6357,CN1CCc2cc(C(N3CCN(C(=O)C4=CCCCO4)CC3)=O)sc2C1 6358,c1(C(=O)NC2(CC=C)CN(c3ncns3)C2)cn(C2CC2)c(C)cc1=O 6359,Cc1ncnc(C)c1C(=O)NC1C(C(=O)NCCc2cnn[nH]2)C1(C)C 6360,c1(CNC(c2ccc(OCCCC)nc2)=O)ccc2cccc(Br)c2n1 6361,c1(C(=O)NCC(COC)O)oc(CNC(C2CCCS2)=O)nc1C 6362,CC1CCC=C1C(=O)NC1(C(=O)NC(CCO)C2CC2)CCSC1 6363,CC1CN(C(c2nccnc2C(N)=O)=O)CC1NC(C1C2CCCC12)=O 6364,c1(NCc2ccc(C(=O)OC)[nH]2)ccc(NC(C2CC2c2ccco2)=O)c(F)c1 6365,Cc1cc(-c2cn(CC(F)(F)CNC(=O)C(C3CCOCC3)F)nn2)ccc1F 6366,Cc1cc(C(C)NC(c2ncsc2Br)c2nnnn2C2CC2)no1 6367,N1(C(c2cccc(-n3cc(C4CCCCCC4)nn3)n2)=O)C2CCCC1CC(O)C2 6368,C1(C(C)NC(C(F)=C(C)C)=O)CCN(C(c2coc(CO)c2)=O)CC1 6369,C1(NC(CC(C(C)C)O)=O)CCN(C(C23CCCCC2C3(F)F)=O)C12CCCC2 6370,N1(c2cc(C(C)=O)ncn2)CC2(CCCC2NC(=O)CCc2ccc(O)nc2)C1 6371,CCCCC(C)CCC(=O)N(CCCCN(C(=O)CC(C)(C)O)C)C 6372,C1(C(N(C)CCNC(=O)COC(=O)C2CC2)=O)(OCC(F)F)CCOC1 6373,c1(C(N(C(C)C(C)C)CC)=O)cc(CNC(=O)C(C2CC2)OC)no1 6374,c1(C(N2CCC(C)(CNC(C3C(C)=C3)=O)CC2)=O)ccccc1N=[N+]=[N-] 6375,N1(C(CSCCN(CC)CC)=O)CCC(F)C(NC(c2cnccn2)=O)C1 6376,C=CC(O)(C(=O)NC1CCN(C(=O)C(n2ccnc2C)C)CC1)C(F)(F)F 6377,N1(C(C2(CC=C)CN(C(c3cnc(C)cc3C)=O)C2)=O)CCC2CCCC2CC1 6378,N1(C(C(CC)(F)F)=O)CCCC(C)(CNC(c2ccc(Br)c(OC)c2)=O)C1 6379,c1(NC(C2(CCNC(c3n(C)nnc3)=O)CC2)=O)ccc2cnccc2c1 6380,CC(CCCCNC(=O)CN1CC=CC1)NC(=O)CCN(C)CCO 6381,C1(OC)(CNC(C2CC(C)(F)C2)=O)CCN(C(C2COCC(C)(C)O2)=O)CC1 6382,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CCN(C(C(C)(C)SC)=O)CC1F 6383,c1(OC)cc(C(C)NC(c2cccc(-c3cc(C(F)(F)F)n[nH]3)n2)=O)cc(F)c1 6384,C12(C(=O)NC(CC)(CNC(c3cc(C#N)c[nH]3)=O)CC)CC(C)(C1)OC2C 6385,N1(C(c2cc(O)ncn2)=O)CCC2(CC1)CC(NC(=O)CN1CCCCC1)C2 6386,C(CC(C(=O)NC1(C)CC1)NC(C1CC2CCC2C1)=O)N(C)C 6387,C(CCC(C)C)(C(=O)NCC12CC(CCO1)C2)NC(c1cccc(CC)n1)=O 6388,c1(C(=O)NC(C)CCNC(c2scnc2Cl)=O)ccnc(O)c1 6389,c1(NC(C)=O)ccc(C(=O)N(CCCNC(=O)Cc2c[nH]nc2O)CCO)nc1 6390,CS(=O)(=O)C1(C(=O)NCCN2CCC(NC(=O)CC3C=CCCC3)CC2)CCC1 6391,CCCCC(CNC(=O)Cc1cncn1C)NC(=O)CC(C)N(C)C 6392,Cc1nccnc1C(=O)NC1CC(C(=O)NC(C2CCCO2)CO)C1 6393,C1(C(=O)OC)CC=C(C(C(=O)NCC2CCOCC2)N2CCC(C(N)=O)C2)CC1 6394,N1(C(CC(=O)N(C)C)=O)CCC(NC(=O)CN(C)S(=O)(=O)N(C)C)C(CO)C1 6395,N1(C(C(C)C(F)F)=O)CCC(CCN(C)C)(C(=O)N(CCC(F)(F)F)C)CC1 6396,c1(C(N2CCC(NC(C(CC3CC3)OC)=O)C2)=O)c(Br)ccc(F)c1C 6397,CC1Sc2ccc(C(=O)NCC3CN(C(=O)C(C4CC4)C4CC4)C3)cc2NC1=O 6398,C#CC1(F)CN(C(=O)CN(C(=O)C(C)OCC2CC2)C)C1 6399,C1(CNC(=O)C2=CCCC2)CN(C(=O)C2=CSCCO2)CCCO1 6400,C(=O)(CCC(C)(C)C)N1C(C)CC(NC(C(Cc2ccc(C)cc2)N(C)C)=O)C1 6401,Cc1cnoc1C(=O)NCC(C)(O)CNC(c1[nH]cnc1C)=O 6402,C1(C(=O)NC2CCCCN(C(C(C(CC)O)C)=O)C2)CCc2nccn2C1 6403,c1(CN2CCC(CC(=O)N(c3ccc(Cl)cc3)CC)CC2)cccc(OC)c1Cl 6404,C1(F)(CNC(c2n(C)nnc2)=O)CCCN(C(=O)C(C)(C)CF)C1 6405,C1(NC(C=CC=CC)=O)CN(C(=O)Cc2ncc(C)[nH]2)C2CCCC12 6406,C1(NC(C(C)(C2CC2)OC)=O)CCCCC1C(=O)NCCC12CCCC1C2 6407,C(=O)(C(CNC(=O)CC1CC(=O)C1)C(C)C)N(c1cn(CCC)nc1)C 6408,c1(CCNC(c2c(Br)cc(C)c(C)n2)=O)ccc2c(n1)OCCO2 6409,C1(C(N2CC(N(C)CC)C2)=O)CCCC(NC(C2(C#N)CCC2)=O)CC1 6410,C1(CNC(C(Br)=C(C)C)=O)CN(C(C2CC2c2cncn2C)=O)CCCO1 6411,c1(CNC(CC2N(C(C(C)n3cccc3)=O)CCC2)=O)ccc2nc[nH]c2c1 6412,C(CCN=c1nc2c(c[nH]1)COC2)NC(=O)C=Cc1cnc[nH]1 6413,C(=O)(C(C)(C)Cc1ccc(O)cc1)NCC(CNC(c1n(CC)nnc1)=O)OC 6414,Cc1cc(C(N2CCCCC2CNC(C2CC(F)C2)=O)=O)sc1Cl 6415,O=C(N=c1[nH][nH]c2c1CN(C(c1c(O)cccc1Cl)=O)C2)c1nc(Cl)ccc1Cl 6416,N#CC1=C(C(=O)NCC2(O)CCN(C(C34CCC(CC3)CO4)=O)C2)CCC1 6417,C(C(O)CC(=O)NC1CCCC(NC(=O)CSc2nc[nH]n2)C1)N(C)C 6418,N1(C(c2nc(OC)oc2)=O)CC2CC3CC2C1C3NC(c1cc(C)oc1C)=O 6419,Cc1[nH]c(C#N)cc1C(=O)NCCC1CN(C(C2CCCOC2C)=O)CCCO1 6420,C(=O)(C(C)C(C)NC(=O)CC1CNC(=O)O1)NCc1c(C(C)(C)C)n[nH]c1 6421,C1(C(N2CC3(C(NC(CCCOC)=O)CCC3)C2)=O)CCC2(CCCC2)CC1 6422,CC(CC(=O)NCCC1CCCOC1)C(C)(C)NC(c1ccc([N+](=O)[O-])[nH]1)=O 6423,S(=O)(=O)(c1cc(F)ccc1OC)NC1CC2(CC(NC(CCC=C)=O)C2)C1 6424,N1(C(C(CO)OC)=O)CC2CCC1CC2NC(=O)CC1CC=CCN1C 6425,C=CC1OCCCC1C(=O)NCCN(C(C1CCCCC1)=O)CC1CC1 6426,C(=O)(CS(=O)(=O)CC(=O)N(C)CCNC(C1CCCC2(CCC2)C1)=O)OC 6427,N1(CC(N2CC3CC(O)CC2C3)=O)Oc2ccccc2S1(=O)=O 6428,C1(CNC(CC(=C)I)=O)C(C)CCCN1C(=O)Cc1cnc[nH]1 6429,C1(N(C(=O)C=Cc2ccco2)C)CCCN(C(=O)CC(O)Cc2ccccc2)C1 6430,C1(C)(CCNC(C(c2ccc(O)cc2)OC)=O)COCCO1 6431,C(CCS(C)(=O)=O)(C(=O)N(C1CCCN(C(=O)COCCC(C)C)C1)CC)OC 6432,CC(CN=c1cc[nH]cc1S(=O)(=O)NCCC1(CO)CCC1)S(N)(=O)=O 6433,c1(C2CN(CC3C(c4n(C)nnn4)CCCC3)C2)cc(-c2ccccc2)ccc1F 6434,CC1=CCC(C(N2CC(COC)(NC(C3CCCC34CC4)=O)C2)=O)CC1 6435,N1(CC)CCC=C(c2cc(C(N3CCc4nncn4CC3)=O)cc3c[nH]nc23)C1 6436,C(CCCCC(=O)NC1CCC(C)(CNC(c2[nH]ccc2C)=O)CC1)=CC 6437,C1(CC)C(C(=O)NC2CC(NC(=O)C=CCNC(=O)OC(C)(C)C)C2)CCN1C 6438,N1(S(c2cc(C(=O)OC)c(Br)cc2)(=O)=O)CCC2(C1)C(=O)NC(=O)N2C 6439,N1(C(C(C(C)O)C)=O)CCN(C2CCCN(C(c3c[nH]ccc3=O)=O)C2)C(=O)C1 6440,C(=O)(CC(C)(C)NC(C1CCC(=O)O1)=O)NC(c1ncn(C)n1)C 6441,c1(C(=O)NC(C(C)NC(c2cccc(C(C)C)n2)=O)CO)cc(Cl)c(F)cc1O 6442,c1(OC(N(C)Cc2cn(C3COCC3OC(C)(C)C)nn2)=O)csc(I)c1 6443,Cc1ccc(F)c(C(N2CC(O)(CNC(=O)C(C)C(C)C3CCCCC3)C2)=O)c1 6444,CC#CCCC(=O)NC(C)(CNC(=O)C(Cc1ccsc1)NC=O)C(C)C 6445,C(C(CC1CC1)C(=O)NCc1ccncn1)NC(C1(C)CC(=O)C1)=O 6446,N1(C(c2c(O)cc(C)nn2)=O)CC(NC(=O)CCn2cncn2)CC12CCCC2 6447,c1(C(=O)NC(CCNC(C)=O)C(C)C)cc(O)nc2c(Br)cccc12 6448,C(=O)(C(O)C(F)(F)F)NC1(CNC(C2CN(C3CCN(C)CC3)C2)=O)CCC1 6449,N1(C(c2ccc(OC)cc2N)=O)CC2OCCN(C(=O)Cc3ccnn3C)C2C1 6450,C(=O)C(C)C(O)CC.C(=O)(CC(OCC)OCC)NCC 6451,N1(CC2C(C3CCC3)C2)CCC(NC(=NCC2CC2)NC2CCOCC2)CC1 6452,C(=O)(CC1COCc2ccccc21)Nc1ncnc(-c2cccc(C)c2)n1 6453,C#Cc1ccc(F)c(C(=O)N(CC)CC2CCCN2C(C2CC(F)C2)=O)c1 6454,C1(NC(Cc2ccc(C)s2)=O)CC2(NC(=O)CCC3(C)CC3)COC1C2 6455,C1(C)(CNC(CC(=C=C)C)=O)CCN(C(=O)CCC2CCCC(O)C2)CC1 6456,c1(C(=O)NCC)cnc2n1CCN(C(c1cc(-c3ccoc3)on1)=O)C2C 6457,c1(C(N)=O)cccc(CNC(C2CC(F)CN2C(C2CNC(=O)O2)=O)=O)c1 6458,N1(C(c2c(C)nccn2)=O)CCN(C(C2OCCCC2(C)C)=O)C2CC12 6459,C1(C(=O)NCC2(C)N(C(C(C)=C(C)C)=O)CCC2)CC2(C1)CC(C)(C)C2 6460,CN1CCOc2c(C(N3CC(CNC(C4(C)COC4)=O)CC3(C)C)=O)cccc21 6461,CC1CN(C(C23CCN(CC2)C3)=O)CCC1CNC(=O)Cn1ncc(Br)n1 6462,c1(NCCSC(C)(C)C)cc(N2CCOC(C3CC3)C2)ncn1 6463,c1(C(N(C)CC)=O)cn2cc(-c3c[nH]nc3C)ccc2n1 6464,CC1CC(C(=O)NCCC2(NC(=O)CSc3nnnn3C3CC3)CC2)CN1C 6465,N1(C(C2(CC#C)CCOCC2)=O)CCC2CN(C(=O)C(C)OCC(F)(F)F)C2C1 6466,N1(C(CCC=CC)=O)CCC(C)C(NC(c2ccc(O)c(C(N)=O)c2)=O)C1 6467,C12(C(N3CC4CC4(CNCc4snc(Cl)c4Cl)C3)=O)CCCN1CCC2 6468,c1(C(=O)NC2CCCN(c3ccccc3F)C2=O)cc2cccc(Cl)c2s1 6469,C1(C(=O)NC2CC(CCNC(c3c(CC)nccn3)=O)C2)CC2(CCC2OC)C1 6470,c1(C(=O)NC2CC(NC(c3cccc(C4CC4)c3)=O)C2)cnn2cccc(Cl)c12 6471,Cc1cn2c(C(N3CC(N(C(=O)CC(O)CC4CC4)C)C3)=O)c(C)nc2s1 6472,c1(C(C)CNC(=O)Cc2ncnn2C)noc(CC2CCCC2)n1 6473,C1(OC)CN(C(=NCCCSC)NCC2CCN(C(C)=O)CC2)CC1OC 6474,C(=O)(CCCCCn1cnnn1)NCCC(C)(C)NC(C1(C)CC1)=O 6475,CCCCCC(O)CC(=O)NCCCC(CCC)NC(c1ccc(Cl)nc1N)=O 6476,C1(c2ccc(OCC)cc2)CCN(C(=O)C(F)C(C)C)CC1NC(=O)C(C)CC 6477,C1(C(N2CCCC2CC(c2cccs2)O)C(=O)NC2CCCC2)CC12CCC2 6478,C(CCC(C)C(=O)NCC1(CC(=O)NC2(CF)CCC2)CC1)OC 6479,N#Cc1cc(S(=O)(=O)NC(C2CC(N)C2)=O)ccc1Br 6480,C(=O)(C1=CC2CCC1C2)N1CCCC(NC(C=Cc2cccc(C)c2)=O)(CO)C1 6481,C12(C(=O)NCC(CC)NC(=O)CCN3CCCS3(=O)=O)CCCC(CO1)C2 6482,Cc1cc(N)c(C(=O)NC2CN(C(C3CCCCNC3=O)=O)CC23CC3)cc1C 6483,c1(C(=O)NC(C)(C)CNC(C2CCc3n[nH]cc3C2)=O)ccc(F)c2ccoc12 6484,c1(C(N2C(Cn3cc(CNC=O)nn3)CCCC2)=O)nccc2c[nH]nc12 6485,CN(Cc1c(Oc2ccccc2)cccc1F)N1CC(Nc2ccccc2)C1 6486,CC1CCCC(C)N(C(C2CCCN2C(C23CC2CNC3=O)=O)=O)C1 6487,C(=O)(C(O)C(C)(C)C)NC1(CNC(c2nccc(CC)c2)=O)CCCC1 6488,c1(C(C)C)nnc2cc(NC3CCN(C(=O)CC4CCCCC4)CC3C)ncn12 6489,N1(C(CN2C(C)CCC2)=O)CCOC2(CCN(C(=O)CC3CNC(=O)C3)CC2)C1 6490,N1(C(C(CC#C)(C)NC(C2CCOC2C)=O)=O)CCOC(C(=C)C)C1 6491,Clc1ccc2[nH]c(=NCC3CCC3)nc(N3CCC(OCC(F)F)CC3)c2c1 6492,CON(CN1CC(=O)N(c2cccc(F)c2)C1=O)CCC(C)C 6493,Cc1cc(C#N)sc1C(=O)NC1(CNC(=O)CC2CC(C)(C)CCO2)CC1 6494,C1(NC(C(C2CC2)OC)=O)CCC(N(C(=O)C(CC#N)c2ccccc2)C)CC1 6495,C1(NC(c2scc(OC)c2)=O)CCS(=O)(=O)C12CN(C(C1(C)CC=CCO1)=O)C2 6496,C(=O)(CCC(C)N(C)C)N(C1CCCC1)CCCNC(c1cc(CC)[nH]n1)=O 6497,C1(CNC(CNS(CC)(=O)=O)=O)CC(N=c2[nH]c3cc(C)nn3c3ccccc23)C1 6498,C1(CC=C)CCN(C(=O)C(CNC(=O)Cn2nccc2C)OC)C1 6499,C1(F)(C(N2CC(C(=O)Nc3cc(C)cc(F)c3)C2)=O)CCCCC1(F)F 6500,C1(CNC(C2(CC=C)CC=CC2)=O)C(C)CCN1C(c1nn(C)nc1Br)=O 6501,Cc1oc(C#N)cc1C(N1CCC(C)(C)C1C(N1CCCC(CO)CC1)=O)=O 6502,c1(OC)ccnc(C(N2CCC(N(C)C(c3cc(Cl)cs3)=O)C(C)C2)=O)c1N 6503,c1(C(=O)NCC2C(CNC(c3c(CC)[nH]c(=N)s3)=O)C2)cscc1S(C)(=O)=O 6504,C(CNC(=O)CN1CCCCC1=O)(C(C)C(C)C)NC(c1c(C)csc1)=O 6505,c1(CC(=O)NCCOCCCNC(CC(CCC)C)=O)ccc2c(c1)CCOC2 6506,C1(NC(N2CC(n3c(C(=O)OCC)ncn3)C2)=O)CCc2ncccc2C1 6507,N1(C(C2C(CC(C)C)C2)=O)CC(F)(F)CC1CNC(c1ncc(F)cn1)=O 6508,c1(OC)c(NC(=O)CCc2cc(OC)cc(C)c2OC)cc(Cl)cc1Br 6509,C=CCC(C)(C)C(=O)NCC(C)(C1CC1)NC(c1nccnc1N)=O 6510,N1(C(c2cc(C)sc2C)=O)CC2CCC1(CNC(c1n[nH]cc1C)=O)CC2 6511,N1(C(c2cc(C)nn2C)=O)CCOC2CN(C(c3conc3C(C)(C)C)=O)CC12 6512,c1(C(=O)Nc2cccnc2)ccnc2ccncc12.C12CN(C1)C(=O)N(C1CC1)C2 6513,c1(C(=O)NCC(C)N(C(C(CC)n2cncn2)=O)C)cn(C)nc1COC 6514,c1(SCC(=O)NC2C(CNC(CN(c3ccns3)C)=O)CC2)nc2ccccc2[nH]1 6515,CCC(C)C(CC(=O)N(CC(C)(C)O)C)NC(c1cccc2ccnn12)=O 6516,c1(CNC(C2CCN(Cc3ncccc3F)C2)=O)ccccc1[N+](=O)[O-] 6517,N1(C(CC(=O)N(C)C)=O)CC2CCCN(C(c3cccc4c3CCC4)=O)C2C1 6518,Cc1noc(C)c1C(=O)NCC(F)CNC(C1(C)CC(C)(C)C1)=O 6519,c1(C(=O)NCC2N(C(C3CC(C)N(C)CC3)=O)CC2)ccc2cccnn12 6520,C(C)(C)(C(=O)NC1CC(CNC(c2coc(CS(C)(=O)=O)n2)=O)C1)N(C)C 6521,N1(CC)CCCCCC(N=c2cc(C)[nH]cc2C#N)C1.N1CC(O)CCC1=O 6522,c1(C(N2CCC(NC(c3cnc(OCC)s3)=O)CC2)=O)ccc(N)c(O)c1 6523,c1(OC)nnc(NCCCCc2cccnc2)cc1N 6524,c1(Nc2nc(C)nc(N3CC4CC(C3)CN(C)C4)c2)cccc2ccc(O)cc12 6525,c1(C(=O)NCC(C)(O)CNC(c2coc(C(F)(F)F)n2)=O)ccc2cc[nH]c2n1 6526,c1(Sc2cc(C#C)n(C3CCCCO3)n2)sc2c(c1F)CCCC2 6527,C(C(C)C(=O)Nn1cccn1)N(C(C1C(C)=CCS1)=O)C 6528,C(=O)(C=C1SCC(=O)N1C)N1C(CN(C(C(CN(C)C)O)=O)C)COCC1 6529,N1(C(COCCCCC)=O)CC(C)CN(C(=O)Cn2cnc(Br)c2)CC1C 6530,CCCC(CCC)=CC(=O)NC1CC(NC(=O)CCCn2cccn2)C(O)C1 6531,C1(C#N)(CCC(=O)NC2CCN(C(=O)OC(C)(C)C)C2)CN(C(=O)CNC=O)C1 6532,c1(CNC(CC)CNC(=O)CC(C)CC(C)C)cc2c(OC)cc(OC)nc2[nH]1 6533,N1(C(CC(=O)NCC)=O)CCC2(CCCC2NC(=O)Cc2nccs2)CC1 6534,c1(C(N2CCC3CN(C(CC4CCN(C)C4)=O)CC32)=O)coc2ccc(O)cc12 6535,c1(OC(C)C)ccc(C(=O)NC2CC23CC(NC(c2c[nH]cc2CN)=O)C3)nc1 6536,C1(CNC(C(C)NC(c2ccoc2)=O)=O)C2CC1N(C(=O)CCC1OCCO1)C2 6537,C1(C(N(CC(C)(C)CNC(=O)Cn2ncnn2)C)=O)CC12CCS(=O)(=O)CC2 6538,CC1CC(C(=O)NC2(C(=O)NC(c3cncs3)C)CSC2)CC(=O)N1 6539,c1(CNS(CCOCCOC)(=O)=O)cc(=NCCO)cc(OC)[nH]1 6540,C12(CNC(CCCCC)=O)CCCC1N(C(=O)C(F)=C(C)C)CCC2 6541,C(C(=O)NC1CN(C(c2cc(O)nn2C)=O)CC1C(F)(F)F)(C(C)C)SCC 6542,N1(C(c2ccc(C(C)=O)cc2)=O)CCC(NC(c2n[nH]c(C3CC3)n2)=O)CC1C 6543,C12(C(N3C(C)CCCC3C)=O)CC(C3CCCC3)(C1)C2 6544,N1(C(C(CCCOC)NC(=O)OC)=O)CCOC2(CCCC2)C1C(=O)OC(C)(C)C 6545,c1(CNC(C(COCC)NC(C=CCC)=O)=O)ncccc1O 6546,Cc1cc(CNC(C)(C)CNC(=O)CC(C)C2CC2)ccc1N1CCOCC1 6547,c1(C(=O)NC(CC)CO)ccc(=NCc2cc(F)ccc2Br)[nH]c1 6548,Cc1ccc(OCC(=O)NC2CC(F)CN(C(c3c[nH]nc3F)=O)C2)c(F)c1 6549,N1(Cc2c(OC)cccn2)CC2(CCC(C(=O)NCCOc3ccccc3)O2)C1 6550,Cc1cnc(C(=O)NC(C)CCN(C)C(C2CC2(C)C(F)F)=O)c(Br)c1 6551,Cc1ccc(C)c(C(=O)NC(CNC(c2cn[nH]c2)=O)C(C)C(C)C)c1 6552,C1(O)(C(C)NC(=O)CNC(N)=O)CCCN(C(C2(n3nccn3)CC2)=O)C1 6553,N1(CCN(C(C2(OC)CCCC2)=O)C)CCN(C(=O)CCS(C)=O)CC1 6554,c1(C(=O)NC(C(C)NC(c2c(C)oc(C)c2C)=O)C)ccc2c(c1)COC2 6555,C1(CCC)CN(C(c2cc(C)n(CCO)n2)=O)CCN1C(=O)C(C)C1(O)CCC1 6556,c1(OCc2cc(NC(N(C(C)C)C(C)C)=O)no2)ncc(Cl)cc1Cl 6557,c1(N2CC(N(C)Cc3ccc([N+](=O)[O-])cc3O)C2)ncnc2ccc(I)cc12 6558,C(=O)(C(CC)NC(=O)Cn1cnc(=N)[nH]1)NC1(CSC)CC1 6559,O=C(C1=NOC2(CCC2)C1)NCC1(C(N2CCC(CCO)C2)=O)CCOCC1 6560,C1(C(N2CC(C3(NC(c4c[nH]nc4C4CC4)=O)CC3)C2)=O)CCC2CCC(=O)N12 6561,C1(O)(CNC(c2cc(I)c(Cl)cn2)=O)COCCC1O 6562,C12(CNC(C(C)N(C(=O)C(C)O)CCC)=O)CC(CO)(CO1)C2 6563,c1(C(=O)NC2CC(O)(CNC(C(C)(C)CO)=O)C2)cccc2c1OCC2 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6777,C(=O)(C1=CC2C=CC(C1)C2)NC1CC2(C(NC(c3n(C)cc(Br)c3)=O)C2)C1 6778,C(CC(=O)NC(CCO)C(F)F)(C(F)(F)F)NC(CN(C(=O)OCC)C)=O 6779,C=CCCCCC(O)CNC(c1ncsc1C(C)C)=O 6780,Cc1ccc(OCC(=O)NCCC2CN(C(C3CCCN3C)=O)CC2C)cc1C 6781,c1(C(=O)NCC(CC)NC(c2cc(Cl)no2)=O)ccc(O)cc1F 6782,c1(C(=O)NC2(CC)CCN(C(=O)C(C)CC(=O)OC)CC2)ccc(S(C)(=O)=O)o1 6783,C=CC(O)C(=O)N1CC(CCNC(c2cc(C(C)(C)C)c[nH]2)=O)C1 6784,c1(C(=O)OC)ccc(S(=O)(=O)N2CCC(N)C2)cc1.c12ccc(cc1)c(=O)[nH]2 6785,N1(C(COC(CNC(CCC=C)=O)(C)C)=O)CC(COC)CC1(C)C 6786,C(CCN=c1[nH]ncs1)NC(C1CC(c2cccc(Cl)c2)(C(F)(F)F)C1)=O 6787,C(=O)(C(C)(C)CC(C)(C)C)N1CC(CC)N(C(=O)Cc2cc(Cl)cc(Cl)c2)CC1 6788,C(CN=C(NCC(=O)NC(C)C)NC1CCN(S(C)(=O)=O)C1)c1ccc(C)cc1 6789,N1(C(c2c(CC#N)cccc2)=O)CCC(C2CC2NC(c2csc(Cl)n2)=O)CC1 6790,Cc1oc2ccccc2c1CC(N1CCC(NC(c2cc(CO)on2)=O)C(O)C1)=O 6791,C(=O)(CS(=O)(=O)CCC(F)(F)F)N1CCCC(NC(N2CCC(C)C2)=O)C1 6792,C(=O)NNc1ncnc2sc3c(c12)CCC3.N1(C(C)C)CCCCC1C 6793,n1(CC(=O)NCCC(C(C)C)NC(C2CCC(C)(C)C2)=O)cc([N+](=O)[O-])cn1 6794,CC(CNC(=O)CSc1ccccc1)(CO)NC(c1cscc1C(F)F)=O 6795,c1(C(=O)OC)cc(Cc2cn(Cc3cc(CO)cc(I)c3)nn2)ccc1Br 6796,N1(C(c2ccn(CC)n2)=O)CCC(O)C(NC(=O)C(C)CSC)C1 6797,CC(C(=O)NC(C1CCN(C(C2CCCN(C(N)=O)C2)=O)C1)(C)C)S(N)(=O)=O 6798,CCCCCCC(=O)NC1CC(CCNC(c2cc(Br)co2)=O)C1 6799,C1(C(C)C)CCC(C)CC1C(=O)NC(CNC(C1(CCO)CC1)=O)C(C)(C)C 6800,CC1(O)CN(C(=O)CCC2CCN(C(=O)CN3CCOCC3)CC2)CCC1O 6801,C(=O)(C1=NOC(C)C1C)NC(Cn1cc(CNC(CSC)=O)nn1)C 6802,CCC(C)C(C(=O)N(CCCC(=O)NC1CCCCCCC1)C)N(C)C 6803,c1(C(N2CC(C)C(C(=O)Nc3cc(S(N)(=O)=O)cs3)C2)=O)csc2ccccc12 6804,C=CCCC(C)NC(C1(CNC(c2occc2CSC)=O)CCC1)=O 6805,c1(OC)ccc(C(=O)NCC2(NC(=O)Cc3ccsc3Cl)CCOC2)cc1OC 6806,C(CCCCC(=O)NCCCN(C)C(C1(NC(N)=O)CCCCC1)=O)=CC 6807,C1(C(=O)NC2(CCCNC(c3n(C=C)ncc3)=O)CC2)OCC2CCCCC12 6808,C1(C(N2C(C)CCCC2)=O)N(C(c2ccco2)=O)CCCC1(C)C 6809,c1(OC)ccccc1C1CC1C(N1CC(NC(C2COCCOC2)=O)C(C)C1)=O 6810,CC1(C)OC(=O)CC1C(N1CCC(C(C)(C)NC(c2cncnc2)=O)C1)=O 6811,C1(NC(C(C=C)O)=O)CCC2(CC1)CC2.C12CCCCC1CNC2=O 6812,C1(NC(C(CC=CC)C)=O)CC2(C1)CC(C(=O)NCC1(CC3CC3)CCC1)C2 6813,Cc1cc2ccc(C(=O)NC(C)CN(C(=O)CCc3ccco3)C)cc2o1 6814,c1(CCC(=O)N(CCN(C(c2c(C)nn(C)c2)=O)C)C)ccc(Cl)cc1F 6815,c1(C(=O)NCCC2CCCCN2C(c2cnc(Cl)s2)=O)cc2cccc(Cl)c2o1 6816,c1(CC(C)(C)CO)nc(CSC2CCCNC2)n(CCCO)n1 6817,CCC(CC(=O)N1CCC(N(C)C(C23CSCC2C3)=O)C1)C1CCC1 6818,c1(C(=O)NC2C3(CN(C(C4C(C)C4)=O)C3)CCC2)coc2c1C(=O)NCC2 6819,C1(NC(C(C)NC(CC)=O)=O)CCCCN(C(=O)CCC=CC(C)C)C1 6820,C1(C)(C(=O)NCCC(C)N(C(=O)CC2C=CCCC2)C)CC(F)(F)C1 6821,C(=O)(C1=C(C)OCCC1)N1C(CCC)CN(C(=O)CC2CC2(C)C)CC1 6822,c1(CC(=O)NCCCN(C(=O)CSCc2ccccc2Cl)C)ccc(O)nc1 6823,CC1CCN(C(=O)CCOC2CN(C(c3ccc(C(N)=O)[nH]3)=O)C2)CCS1 6824,c1(C(=O)OC(c2c(OC)cccc2)C2CC2)cc(C)c(O)nn1 6825,c1(C(N2C(C(=O)NCCc3c(C)[nH]nc3O)CCC2)=O)ccc([N+](=O)[O-])cc1Br 6826,N1(C(C=Cc2cn(C)nn2)=O)CCC(NC(c2cc(C3CC3)nn2C)=O)C12CC2 6827,CCCCCCCCCC(=O)NCCN(C(=O)CC(C)(C)C(=O)OC)C1CC1 6828,C1(C(N(C2(C(=O)OC)CC2)C)=O)CC2(CC2)CN1C(=O)C=Cc1ccn(C)c1 6829,C1(NC(c2c(OC)noc2C)=O)CCCCN(C(=O)CC(C)c2cccnc2)C1 6830,C(C1C(C(=O)NCC2(F)CC(NC(=O)COCC(C)(C)C)C2)C1(C)C)=C(C)C 6831,C1(F)(C(N2CC(C)(CC)C2)=O)CCCN(C(c2ccc(Cl)cn2)=O)C1 6832,C1(C(N2CC(C)C(CCNC(=O)C(F)(F)C(F)F)C2)=O)CCCCC1(F)F 6833,C1(O)(CC(=O)NCC(CNC(c2c(C)nc(C3CC3)[nH]2)=O)(C)O)CCCCCC1 6834,C1(COC)(NC(c2cnc[nH]2)=O)CCN(C(=O)C=CC=C(Cl)Cl)C1 6835,c1(OCC(=O)NCC2CCCN2C(=O)CC23CCCC2C3)ccc(C(F)F)nc1 6836,c1(SCCC)ccc(C(=O)NC2CCC(NC(C3CC(CC(F)F)C3)=O)C2)cc1 6837,C(=O)(C1=CCCCC1P(C)(C)=O)NCC1N(C(C=CCOC)=O)CCC1 6838,CCC(CC(=O)N1CCCC(N(C(=O)CCCc2cccs2)CCF)C1)OC 6839,N1(C(=O)NCC2CCC=CO2)CC2CC1C1CC21 6840,CC1COC(C(=O)NC2CCN(CC(=O)Nc3cn(-c4ccccc4)nn3)C2)C1 6841,c1(C(=O)NC2CCN(C(C#CC3(C)CC3)=O)C23CCC3)ccc2c(c1)CCC=C2 6842,c1(C(=O)NCc2cccc(C(N(CC(C)C)CC)=O)n2)cccc2ccoc12 6843,n1(C2CCN(C(c3ccnc(N4CCNCC4)c3)=O)C2)ncc2c1CNC2 6844,c1ccc(Cl)cc1.c1(NC(C)C(=O)NC2(CNC3(CS)CC3)CC2)ccccn1 6845,C(=O)(CCCCC(C)(C)C)N(CC(CC)NC(c1cncc(OC)n1)=O)C 6846,n1(CCC(=O)NC(CNC(c2c(C)ocn2)=O)C(C)C)c(C)cc(O)cc1=O 6847,CCCCCC(C)(C)C(=O)NCCCCN(C(=O)CC(c1cccc(F)c1)O)C 6848,c1(N2CCC(CC(=O)NCCC=C)C2)cc(OC)nc(OC)n1 6849,C1(NC(c2nc(COCC)sc2)=O)C=CCN(c2nccc(CO)n2)C1 6850,N1(C(C2CC(NC(C(C)OCCCC)=O)C2)=O)CCC2(CCCN2C)C1 6851,C1(CNC(c2cc(O)ncc2Br)=O)CCCN(C(c2cnc[nH]2)=O)CC1 6852,C1(COC)(NC(c2cc(Cl)c[nH]2)=O)CCN(C(=O)Cc2ccc(F)cn2)CC1 6853,c1(C(=O)NC(C(C)(C)NC(c2cc(COC)on2)=O)C)ccc2c(c1)CCCS2 6854,N1(C(CN(CCC)C)=O)CC(NC(C2(O)CCSC2)=O)CC2(CC2)C1 6855,N1(CC)C(=O)CCC1C(=O)NC(CNC(c1cc(CO)oc1C)=O)C(C)C 6856,C(=O)(CS(=O)(=O)C(C)(C)C)N1CCC(NC(c2cccc(OC)c2C)=O)C2C1C2 6857,c1(C(=O)OCC)ccc(S(=O)(=O)N2CCC(N)(COC)C2)c(F)c1 6858,C1(NC(CCC)=O)CCNC1=O.C(C(=O)OCC)SC1CC1C(C)C 6859,N1(C(CNC(CNC(C)=O)=O)=O)C2CCC1CC(N(C)C(C1CCCOC1)=O)C2 6860,N1(C(N2CC(C(Cn3cc(-c4cnc(OC)s4)nn3)F)C2)=O)CCC(OC)CC1 6861,c1(C(c2ccsc2)N(CC(C)N(C(=O)C(C)O)C)C)ccc2ccccc2c1 6862,C1(CC)CN(C(=O)C(CCOC)OC)CC1NC(=O)CC=C(C)C 6863,c1(C(=O)NCC2(CNC(CC(=C=C)C)=O)CCOCC2)ccc(Cl)c(CC)c1 6864,C1(CC(=O)NC(C(=O)NCc2nc(CC)[nH]n2)C2(O)CCC2)C=NN(C)C1=O 6865,N1(C(C2(C#N)CC=CC2)=O)CC(NC(C2CC(F)(CO)C2)=O)C(N=[N+]=[N-])C1 6866,CCC(CCO)NC(=O)NCC(c1cnn(C)c1)(C)O 6867,C1(NC(c2c(CC)onc2)=O)CCCN(C(=O)CCc2cc(F)ccc2F)CC1 6868,N1(C(C2(C)CCC2)=O)CCOCC2(C1)CN(C(=O)CC1CCCC1(F)F)CCO2 6869,C1(C(=O)NCC(=O)OCC=C)CC2CCC1N2C(C1CC(=O)C1)=O 6870,N1(C(c2cn(CC)nn2)=O)CCCN(C(=O)C2=CCCOC2)CC1C(C)C 6871,C(=O)(C1=CCN(C)C1)N(CC(CNC(C=Cc1c(C)n[nH]c1)=O)(C)C)C 6872,C(=O)(CC(C)CC(C)(C)C)N1C2(C(=O)NC(CCCC)(C)CO)CC(C1)C2 6873,c1(CNC(=O)Nc2cnn(C(F)F)c2)nnc(CO)o1 6874,C1(C)(CNC(C(CC)F)=O)COCCN(C(=O)CCCCCN(C)C)C1 6875,C(C(CNC(c1ccc([N+](=O)[O-])[nH]1)=O)C(F)(F)F)NC(C1N(CC)CC1)=O 6876,Cc1ccc(C(C)(F)F)cc1NCc1cc(F)ncc1F 6877,C(=O)(C(C)C(C)S(C)(=O)=O)NC1(CCNC(c2ccn(CCC)n2)=O)CCCC1 6878,CCCC(C(=O)NCCCC(C)(C)NC(=O)COC1CCCCC1)NC(C)=O 6879,Cc1ccc(C(=O)NC2CCC(C(=O)Nc3cc(F)cnc3C)OC2)c(O)n1 6880,NS(=O)(=O)C1(C(=O)NC2CC(NC(=O)C=Cc3cocn3)C23CCC3)CCC1 6881,CN1C(=O)CCC1C(=O)NCC1CCCCC1NC(c1cccc(C2CC2)c1)=O 6882,CC(CCCCN=c1[nH]cc2ccnc-2[nH]1)NC(c1cc(C(F)F)on1)=O 6883,N1(Cc2nc(CCCC)sc2)CCC(CNCC(=O)CN2CC3C=CC2C3)CC1 6884,CC1CCCC1N=c1[nH]c(N2C3CCC2COC3)nc2c1CCCC2 6885,C1(C(=O)NC2CC2)C2C3CC4C1C2C34C(N(C)Cc1ccc(C)cc1)=O 6886,C(=O)(CCC(O)C(C)(C)C)NCC(C)NC(C1(C)CC(F)(F)C1)=O 6887,C12CCN(CC1)C2.N1(CC=CC(=O)NC(N)=O)CCOCC1 6888,c1(C(=O)NC(CNC(c2c(C#N)ccs2)=O)CO)cccn2c(O)nnc12 6889,N1(C(CC(C)F)=O)CCC2(CC(C(=O)Nc3ccccc3C3CC3)C2)C1 6890,C1(COC)(Cc2ccccc2)CCCN(C(=O)Cc2c(C)nn(C(C)C)c2C)C1 6891,c1(C(N(CCCNC(=O)C(C)C(F)F)CCC)=O)cccc2ncnn12 6892,C(C(=O)NC1CCN(CC(=O)Nc2cccc(C)c2)CC1C)(C(C)(C)C)OC 6893,CC1(C)C(C)(C(=O)NC2CCC(NC(=O)CC(=O)NC3CC3)C2)C1(C)C 6894,Cc1cc(=NCC2CC(NC(=O)C3COc4ccccc43)C2)[nH]c(S(C)(=O)=O)n1 6895,C(C(CC(=O)NCC(C)C(=O)OC1CC1)C1CCC1)NC(CN(CCOC)C)=O 6896,C1(N(C(C2C(C)OCC2)=O)C)CN(C(=O)C=Cc2ccc(O)cc2)CC1(C)C 6897,C(CC(N)=O)(C(=O)N1CCNC(=O)C1)NC(C1OCCN(C)C1)=O 6898,C1(C(N)=O)(C(=O)N)CC2CCC1C2.C1(O)(CC)CN(CCCc2nn[nH]n2)C1 6899,CC1COCC(C(=O)N(C)CC=CC(=O)NC2CCCC(O)C2)O1 6900,N(C1CCC2(CC2)c2cc(Br)ccc21)Cc1cc2ccc(O)cc2cc1 6901,c1(SCC)cc(Cl)ccc1C(=O)NC1CCC(NC(=O)C(C)n2cccc2)CC1 6902,N1(C(C2C(NC(c3cccc(-c4ccccc4)c3)=O)C2)=O)CC(O)C(O)C1 6903,CC1(C)CC(C)(C(N2CCC3(CCC3)C2)=O)CN1C(=O)CC#N 6904,N1(C(c2c(CN(C(=O)C(C)SC)CC=C)cccn2)=O)CC(F)(F)CC1(C)CO 6905,C1(NC(c2c(C)nccn2)=O)CCCC12CCN(C(=O)C1=CCS(=O)(=O)C1)C2 6906,Cc1nc(S(=O)(=O)N(C(=O)C(F)CC(C)C)C(C)C)ccc1Br 6907,C(=O)(C1=CCCCCC1)NC1CC(F)(CNC(=O)CC2CCCNC2=O)C1 6908,CCCCCC(O)CC(=O)NCC(C)N(C)C(c1ccnc(F)c1Cl)=O 6909,C1(NC(C2N(C)CC(C)(C)C2)=O)CCC2CC1CN2C(=O)C1=CCOCC1 6910,C(CCCCCNC(=O)C(C1CCN(C(=O)C(CO)NC(N)=O)C1)F)N(C)C 6911,N1(Cc2c(C(S(C)(=O)=O)NCCC)cccc2)CCCC2(CCCO2)C1.c1ccccc1 6912,c1(NCC)ccc(Cl)c(C(=O)NC2(n3cc(C#N)cn3)CC2)c1 6913,CC(C)(CCC(=O)NC1CCC(NC(c2cnc(N)cn2)=O)CC1)[N+](=O)[O-] 6914,CC1(C)CCC(C(=O)N(CCNC(=O)C(c2cccc(F)c2)O)C2CC2)OC1 6915,N1(C(c2c(NCCCC)ccc(Cl)c2)=O)CCCC2(C1)CC(F)(F)C2 6916,C1(NC(CN2CC(=O)N(C)C2=O)=O)CCCCCN(C(=O)Cc2ccsn2)C1 6917,Cc1cc(N)c(C(=O)NC2CC(CNC(c3cn(C)c(O)n3)=O)C(O)C2)c(F)c1 6918,c1(CCC(=O)NC(C(C)NC(c2c(CC)nccn2)=O)(C)C)c(C)nn(C)c1C 6919,N1(C(C2(C(C)NC(C(C)SCC)=O)CC2)=O)Cc2c[nH]nc2C1 6920,C12(NC(C3CCCCC3)=O)CCCC1N(Cc1cscn1)CC2 6921,c1(CC(=O)NCCCCC2CCCN(C(C(C)(C)O)=O)C2)cccc2nsnc12 6922,C1(C(=O)NC(CCN(C(COCC)=O)C)C(C)C)CC2(C1)C(F)(F)C21CC1 6923,N1(C(C(C2CCCC2)OC)=O)CCC(NC(=O)C(N)=O)C(C)(C)C1 6924,C1(NC(C2COCCN2CC(F)F)=O)CN(C(c2cncc(Cl)c2)=O)CCC1O 6925,C1(C2CC2)(NS(N(C)CCOC)(=O)=O)CCCCCC1 6926,C1(CNC(c2n(C=C)ncc2)=O)CCN(C(c2ccc(F)cc2C)=O)CC1C 6927,N1(C(c2n(COC)ncc2)=O)CCOC(C)C1C(N1CC2(CO)CC2(CO)C1)=O 6928,C(CC(=O)NOCCOC)(C(F)(F)F)NC(C1(CC=C)CCCC1)=O 6929,c1(C(=O)OCC(CC(C)C)F)ccccc1S(=O)(=O)C(C)C 6930,N1(C(c2c(C)nn[nH]2)=O)CCN(C(c2ccc(Cl)s2)=O)C(C)C1C 6931,CC1CCN(C(=O)C(O)Cc2cn(C)cn2)C(CNC(c2cnccn2)=O)C1 6932,N1(Cc2ccc(CC)cc2)CCN(C(C2CCN(C)C2)=O)CC1c1nccn1C 6933,CC1(C)CCC(NC(C2COCC2CNC(=O)CC2CC3CCC2O3)=O)CC1 6934,C1(NC(C2C(C)C2C)=O)CN(C(=O)CC2CC3(CCO2)CC3)C2(CCCC2)C1 6935,Cc1ccc(NC(=O)CCCCNC(c2ccccc2CC#N)=O)cc1O 6936,C(=O)(C(C)(C)COC)NCC(CC)NC(c1cccc(F)n1)=O 6937,C(=O)(CN=c1cc[nH]cc1)NCCOCCC(=O)NC(C)CCn1cncn1 6938,Cc1cnc(O)c(NC(C2(O)CCN(Cc3ccc(Br)c(O)c3)C2)=O)c1 6939,N1(C(CCCC(C)c2cn(C(C)C(=O)O)nn2)=O)CCC2COC(=O)NC2C1 6940,C(=O)(CC1CCOc2ccccc21)N(C(CCNC(CC(=O)NCC)=O)C)C 6941,c1(OC)cc(C(=O)NCC=CCC(=O)N(C)CCc2cnccn2)n(C)n1 6942,CC1CN(C(C2CC3(CC(NC(C4C=CCC4)=O)C3)C2)=O)CC(C)(C)O1 6943,N1(C(CCCCOCC)=O)CCN(C(=O)CCC(C)N(C)C)CC1CC(F)(F)F 6944,C1(NC(COCCC)=O)(COC2(C)CCOC2)CCCC1 6945,C(=O)(C(O)C(C(C)C)OC)N1CC(CC)C(NC(c2cc(C)ncc2Cl)=O)CC1 6946,C(C)(C(=O)OCCC(=O)N(C)C)N(C1CCCC1)C(CNC(C)=O)=O 6947,C1(F)(C(=O)NCC2(CNC(c3c[nH]nc3F)=O)CC2)CCOCC1 6948,CN1CC(O)CCC1C(=O)NC1C=CC(C(=O)NC2(CO)CCC2)C1 6949,Cc1cccc(OCC(=O)NC2CN(C(c3cnsc3)=O)CC2O)c1F 6950,CN(C)S(=O)(=O)N1CCC(CN2CC3(CCC3)C2c2ccsc2)CC1 6951,S(=O)(=O)(c1cccc(Cl)c1)NC(C1C(C(N2CCCNCC2)=O)C1)=O 6952,CC1(C)CCN(C(C2(O)CCCCC2)=O)CC1CNC(c1c[nH]nc1Br)=O 6953,C1(CN(C(=O)C(O)COC)CC)CCCN1C(c1cnn(C(F)F)c1)=O 6954,N1(C(CCOCCOC(C)(C)C)=O)CCC(NC(=O)C=CC(F)(F)F)C1 6955,c1(-c2nc(C(C)C3CC3)nn2C2CCCOC2)ccnc(O)c1Br 6956,c1(OC)c(Cl)cc(NC(C2CC(O)CN2S(=O)(=O)c2cccs2)=O)cc1Cl 6957,Cc1cnc2n1CCCC2C(=O)N1CCN(C(C2CS(=O)(=O)C2)=O)C(CO)C1 6958,CC(C)C(N=[N+]=[N-])C(=O)N1CCC(C)(CCNC(c2ncn3ccccc23)=O)C1 6959,C(C)(CNC(=O)CCc1ccc(Br)s1)(CC(C)C)NC(CC(C)C)=O 6960,Cc1ccc(C(N2CC(F)(C(N3CCN4CCOCC4C3)=O)C2)=O)c([N+](=O)[O-])c1 6961,c1(CC(C(=O)N(CCC)CCNC(=O)Cc2csc(S)n2)C)c(C)n[nH]c1C 6962,N1(C(C(C2CCN(C(c3ccnc(O)c3)=O)CC2)C)=O)CCc2ncccc2C1 6963,C1(O)(CN(C(C(CC=C)C)=O)C)CCCN(C(c2cnc(C(C)(C)C)o2)=O)C1 6964,C(=O)(CCC(C)(F)F)NC(CC(=O)NC1(C#C)CC1)COC 6965,CC(C)(C(=O)NC1CCCC1NC(=O)CCOCc1ccccc1)C1CCCO1 6966,c1(NC(C)CNC(=O)C(F)(F)c2cncs2)ncc(F)cn1 6967,Cc1[nH]nc(C(N2CCCN(C(=O)CCCSC(C)(C)C)CCC2)=O)c1[N+](=O)[O-] 6968,n1(CCCC(C)O)cc(C#CCN(C(N)=O)NC(=O)CNC(=O)OC(C)(C)C)nn1 6969,N1(C(c2ccc(C3C(C)C3)o2)=O)CCC(F)(CNC(=O)C(O)CC(N)=O)CC1 6970,C1(NC(=O)NCC2(CCOC)CCC2)CCC(C)c2ccccc2C1 6971,CC1CC(F)(F)CN1C(C1(NC(=O)C(O)C2CCCC2)CCSC1)=O 6972,CC(C)C(F)(CNC(=O)C1=CCCC1C)C(=O)NC(C)(C)CNC(N)=O 6973,c1(OC)cc(N2CCC(NC(C3(C4CCOCC4)CC3)=O)C2)c(F)cc1[N+](=O)[O-] 6974,C1(C(=O)NCC2(OC)CCCCC2)CN(C)CCN1C(c1cc(C)n(C)c1C)=O 6975,C1(C(N(CC(CN(C(C2(SC)CCC2)=O)C)O)C)=O)CC(C)(C(C)(C)C)C1 6976,C1(NC(C(C(=O)OC)C)=O)CC(F)(F)CC1NC(c1conc1C)=O 6977,N1(C(c2ccc(C#C)cn2)=O)CC2(CCN(C(=O)C(C)(CC)CO)CC2)C1 6978,Cc1ccc(F)cc1CN(C(=O)C(=O)NC1(Cc2cc(=O)n(C)cn2)CC1)C 6979,O=C(CCC(=O)NC1C(NC(c2ccns2)=O)CCOC1)Nc1cccs1 6980,N1(C(c2c(C)nns2)=O)CC(NC(c2occc2F)=O)CC(O)C1 6981,Cc1cc(C(=O)NCC(=O)NC2COCCC2NC(=O)CC2CCCO2)n(C)n1 6982,c1(OC)c(C(=O)NC(C)(C)CCCNC(C2CCC(=O)O2)=O)cc(F)cc1F 6983,C1(C)(CNC(C(C)SCc2cccc(C)c2)=O)CN(C(=O)C(C)(F)F)CCO1 6984,Cc1c(F)ccc(F)c1CN1CCC(O)(CC(N2CCCOCC2)=O)CC1 6985,N1(Cc2onc(CC)n2)CCC(CO)(NC(C2CCCN2C(C)=O)=O)CC1 6986,Cc1c(Cl)ccnc1NNC(=O)N1CCCCC1c1cccnc1O 6987,n1(CC)nc(C)cc1C(=O)NC1C=CCN(C(c2ncoc2Br)=O)C1 6988,c1(CCC)c(C(N2CCC2CNC(c2nccnc2N)=O)=O)nnn1CC 6989,C1(CNC(C2C3(CCN(CC(=O)OCCC)CC3)C2)=O)CCC2(CCCC2)CC1 6990,n1(CC(=O)N(CC(CN(C(=O)CC2C=CCCC2)C)O)C)ccc(Br)n1 6991,c1(C(N2CC(NC(CCOC(C)=O)=O)C2)=O)cc(F)c(Br)cc1F 6992,N1(C(CC2(OC)CCCC2)=O)CCN(C)CC1CNC(=O)CC(C)CN(C)C 6993,C1(C(=O)NC(C2CCCC2)CC)CN(C(c2[nH]ccc2C2CC2)=O)CCN1C 6994,c1(CC(=O)NCC(C)N(C(=O)CC2CC(=O)NC2=O)C)c[nH]c2c(F)cccc12 6995,Cn1cc(Br)cc1C(N1CC2CC2C1CNC(=O)CCn1cncn1)=O 6996,C1(c2n(-c3c(SC)cccc3)nc(-c3cncnc3)n2)CC(=O)NC1(C)C 6997,c1(C2(NC(=O)NCC(F)C3CNC3)CCC2)ccccc1 6998,C1(CNC(C=CCOC)=O)CCN(C(c2ccc(F)cc2Br)=O)C1(C)C 6999,C(C(CC)CC(C)C)NC(C(=O)NC(CC#CC)C)=O.C1CN1 7000,C1(C(N)=O)CCC(C(=O)NC2CC(F)(CNC(=O)CC3COCCO3)C2)CC1 7001,C1(NC(Cc2cc(C)c(Cl)cc2)=O)COC2C(NC(C3(C)CCCC3)=O)COC12 7002,c1(OC)cc(CCO)ccc1Nc1ccc(N2CCCC2)nn1 7003,N1(C(C2N(C)CCN(C(c3cc(CC)[nH]n3)=O)C2)=O)CC2(COC(=O)N2C)C1 7004,C(=O)(C(O)CCCNC(C1CCCSC1C)=O)NCc1cc(C)ns1 7005,CC(CCP(C)(C)=O)(c1nnnn1C1CCC1)NCCCCn1cnnc1 7006,N1(C(C(CC(C)C)N(C)C)=O)CCCC(NC(c2cn[nH]c2)=O)CCC1 7007,c1(COC(C(C)(C2CCC2)NC(C(CC2CC2)OC)=O)=O)ccc(Cl)nc1 7008,N(C(=NCC1COCCO1)N1CCN2C(=O)OCCC2C1)C1(C)CCCC1 7009,C(C)(CN=c1[nH]ccc2cccc(C)c12)(CC(C)C)OCC 7010,C1(C(=O)NC(C2CCCC2)C#C)CCCN1C(C1CCCSC1)=O 7011,C=C1CC2CCC(C1)N2C(=O)C(C(C)CC)N(C)C(c1ncc(F)cc1F)=O 7012,c1(OC)cc(CN2CCOC(C(=O)NCc3ccn(C)n3)C2)ccc1C 7013,CC1CC(NC(c2ccccc2-n2cncn2)=O)CN1C(=O)CC1(C)CCCC1 7014,Nc1cc(C(N2CC(F)(CNC(C3C(F)(F)C34CC4)=O)C2)=O)c(F)cc1F 7015,C1(CNC(CC(CC)OC)=O)CCC2(CCC2)CN1C(C1CC1C1CCC1)=O 7016,C1(NC(C2CCCC(=O)N2)=O)CCN(C(c2cnc(C(F)(F)F)s2)=O)CC(O)C1 7017,N1(C(C2N(CC)CCC2)=O)CCN(C(c2c(Cl)cnn2C)=O)CC1CC(=O)NC 7018,c1(CN2CC(C)C2Nc2ncc(C(F)(F)F)cn2)ccc2sccc2c1 7019,c1(NC(c2ccc(C(=O)OC)s2)=O)cc(OC(N2C3CCC2CC3)=O)n(C)n1 7020,CC1(C)CN(C(c2sccc2Cl)C(=O)NCc2cccc(OCCO)c2)CC1CO 7021,C(=O)(C(C1=NOC2CC12)N(C)Cc1ccc2c(c1)OCO2)NCCCOC 7022,N1(C(C(=O)NC2CC3(CC(OC)C3)C2)=O)CC2(CCC2)CC1CO 7023,Cc1cnoc1C(=O)NC(C)(CNC(C1CCN(C(N)=O)C1)=O)C1CC1 7024,N1(C(CC(CC)SC)=O)CCC(CNC(c2cnc(O)c(F)c2)=O)C(O)C1 7025,C12(NC(C(C)CN(C)C)=O)CCOC(CNC(c3ncccc3C(F)F)=O)(C1)C2 7026,c1(C(N2CCC(CCN(C(C(CC)OC)=O)C)CC2)=O)cc(F)c(Cl)cc1F 7027,c1(CCNC(=O)NCCc2ccc(N3CCN(C)CC3)cc2)c(F)cccc1F 7028,c1(CNC(c2c(NC(CC(=O)OC)=O)ccs2)=O)ccc2c(c1)COC2 7029,C(CS(=O)(=O)CC(=O)NC1CCCN(C(c2cc(C)co2)=O)C1C)OC 7030,N1(C(CN2CCC(C)(O)C2)=O)CCN(C(=O)C(C)(C)O)CC12CCC2 7031,c1(CC(=O)N(C)CC2N(C(CCCCSC)=O)CCC2)cccc(F)c1O 7032,C(CNC(C1C2COCC12)=O)(CC(F)(F)F)NC(c1c(SCC)nccn1)=O 7033,C(=O)(C(C)CS(C)(=O)=O)N1CCC(NC(c2sc(CC)c(C)c2)=O)C1 7034,CC(C)(C(=O)NCCCCNC(C1(c2ccc(Cl)nc2)CC1)=O)C(F)(F)F 7035,N1(C(CSCCCC)=O)CCOCC(F)(CNC(=O)C=Cc2cnc[nH]2)C1 7036,CCC(C)(C#N)C(=O)NC1(CC(=O)NCc2cnn(CCF)c2)CC1 7037,S(=O)(=O)(c1ccc(C(C)(C)C)cc1)N1C(C(=O)NC(CN(C)C)(C)C)CCCC1 7038,C1(C)(C(=O)NC(CCCNC(c2ccc(SC)o2)=O)C)CC=CCO1 7039,C1(CNC(c2cncs2)=O)CCCN(c2cc(-c3ccccc3)ncn2)C1 7040,N1(C(CC(C)OC)=O)CCC2(CC1)CN(Cc1ccc(Cl)cc1C)CCO2 7041,c1(NCC(=O)OCc2ncccc2Cl)ccccc1Cl 7042,C1(NC(C2CCCS2)=O)CCSC12CN(C(=O)CCc1nc3ncccn3n1)C2 7043,CC#CCCCC(=O)NCC1C=CCN1C(c1ccc(CCC)c(N)c1)=O 7044,c1(N(C)Cc2cccc(OCF)c2)nc(N2CCC(S(C)(=O)=O)C2)c2c(n1)COC2 7045,Cc1cc(=NCC2CC2(C)C(F)F)[nH]c(C(c2cc(C)oc2C)C)n1 7046,n1(CC)cc(CC(=O)NC2(CCNC(C3CC(CC(F)F)C3)=O)CCCC2)cn1 7047,c1(CN(C(C)C)C(=O)Nc2cccnc2Oc2ccccc2)cc(Br)ccc1F 7048,Cc1onc(C(=O)NC2CC2CNC(=O)CSc2ccccc2)c1Br 7049,C1(OC)CC2(C1)NC(=O)N(C1CCCC(C)C1)C2=O 7050,c1(OC)cc(C(F)F)c(C(=O)NCC(C)N(C(=O)Cn2cncn2)C)cn1 7051,C(=O)(CC(C)CC(=O)NCC1C(CC2(C(=O)NN(C)C)CCC2)C1(F)F)OC 7052,Cc1oc(C)c(C(=O)NC(C2CCN(C(=O)Cc3cccc(O)c3)C2)C)c1C 7053,C1(C(=O)NC2CC(N(C(CSCCCC)=O)C)C2)CCc2nc(O)[nH]c2C1 7054,c1(NCC(=O)NC2(CNC(=O)CSC3CCCCO3)CC2)cccnc1 7055,Cc1nn(C(F)(F)F)c(C)c1CN(C1CC2CCC1CC2)C 7056,C1(CC=C)(NC(c2cc(C(=O)OC)c[nH]2)=O)CCCN(C(C2CCCC2)=O)C1 7057,C1(CNC(c2scnc2Cl)=O)CN(C(C2CN=C3N=CNN3C2)=O)CCC1(F)F 7058,c1(CN2C(C(N3CCC(F)(F)C3)=O)CSCC2)cnc(Cl)cc1Cl 7059,C1(C(=O)NCC(n2cc(CCN3CCC(O)CC3)nn2)C)CCCC2NCCC12 7060,C1(CCNC(C(c2n(C)ncc2)(F)F)=O)CN(C(c2ccsn2)=O)CCO1 7061,Cc1cnncc1C(=O)NCC(C)(C)CN(C(=O)COCC(=O)N(C)C)C 7062,N1(C(C(CC)=CC)=O)CCOC(C(C)NC(c2ccc(Cl)cn2)=O)C1 7063,c1(CCNC(=O)NC(CC(=O)OC)C2CCCCC2)nccc(C(F)(F)F)n1 7064,N1(CC)CC(C(=O)N(C)CCC2CCCCN2C(=O)CCSC)CC1=O 7065,C(=O)(CC(C(=O)NC1(C)CN(C(c2scnc2C(C)C)=O)C1)N(C)C)OC 7066,C1(C(N2CCC(NC(C=NOC)=O)C2(C)C)=O)CCc2nccn2C1 7067,N1(C(C=CCOCCOC)=O)CCC2C(NC(C3CC(CO)(CO)C3)=O)C12 7068,C#Cc1ccc(C(N2CCC(c3n[nH]c(CNC(=O)C(O)C(C)C)n3)C2)=O)nc1 7069,C(=O)(C1CCc2c[nH]nc21)N1CC(C(C(=O)NC(c2cnccc2Cl)=O)OC)C1 7070,C1(CCCCC)CCC(C(N2CCN(C(=O)CC3CCCCO3)CC2)=O)CC1 7071,CN1CCN(C(c2coc(CNC(=O)C=Cc3cccc(F)c3)n2)=O)C(CO)C1 7072,C(c1cccc(C(F)(F)F)c1)=CC(=O)N(C1CN(C(C(F)OC)=O)C1)C 7073,C1(NC(c2cnc(C(C)OC)s2)=O)CCN(C(=O)C(C)(C)NS(C)(=O)=O)CC1F 7074,Cc1cc(C)c(C(N2CCC(CNC(c3cc([N+](=O)[O-])n[nH]3)=O)C(C)C2)=O)cn1 7075,C1(=CC(=O)NCC(CNC(c2nccc(Cl)c2F)=O)OC)CCCCC1(C)C 7076,CCC(C)(CNC(C1CN(S(=O)(=O)CC)C1)=O)NC(=O)C(C)(C)c1csc(C)c1 7077,c1(OC)cc(CC(N2CCN(CCNC(C3(O)CCCC3)=O)CC2)=O)ccc1C 7078,N1(C(C(C)OC)=O)CC2CN(C(c3ccc(C(C)C(F)(F)F)cc3)=O)CC12 7079,c1(C(=O)NC2CN(C(c3cc(C)cc(O)n3)=O)CC2C)[nH]cc2c1CCCC2 7080,C1(C(=O)NCC2C(C(N3C(C#C)CCC3)=O)C2(C)C)CC2COCC2C1 7081,c1(CN2CC(CC)N(c3ncc(Br)c(C)n3)CC2)cn2c(Br)cccc2n1 7082,C(=O)(C(F)(F)C(F)(F)F)NCC(CNC(c1ccnc(C)c1C)=O)(C)F 7083,c1(CC)[nH]c(=N)sc1C(=O)NC1CC(CNC(c2c[nH]cc2Br)=O)CC1O 7084,N1(C(C2C3CN(C(CC4(NC(C)=O)CC4)=O)C2C3)=O)CCCCCCC1C 7085,N1(C(C(C(C)OC)N(C)C)=O)CC(C)(C)CC1CC(=O)N(CC(C)(F)F)C 7086,c1(C(N(CCS)CC)=O)cnc(OCC(O)COC)cn1.C1(C(C2CC2)=O)CCCC1 7087,O(NC(=O)C(c1cccs1)NC(c1coc(CO)c1)=O)CCCC#C 7088,C(C)(C)(CC(=O)NCC(Cl)C(C)(F)F)N(C(CN1CCC(C)C1)=O)C 7089,N1(C(c2scc(OC)c2)=O)CCC2(CCCN2C(C2(O)CCC(C)(C)CC2)=O)C1 7090,c1(NC(c2nccs2)C)nccc(N2CCC(N3CCOCC3=O)CC2)n1 7091,N1(C(C(C2CCN(C(c3cnc(C#N)s3)=O)C2)C)=O)CCOC(C2CCC2)C1 7092,c1(C(C(N2CCC(NC(C(C)OC(C)(C)C)=O)C2)=O)(C)C)cc(Cl)cc(Cl)c1 7093,C(C(CC(C)C)C(=O)NC1CCC1NC(c1cscc1C)=O)OC 7094,c1(C(N2CC(NC(CCc3n(C)cnn3)=O)C3C2C3)=O)cc2sc(Cl)cc2s1 7095,N1(C(c2n(C)ncc2Cl)=O)CCC(NC(=O)Cc2c(O)ncnc2O)CC(O)C1 7096,CCC(O)C(C)(C)C(=O)NC1CCCC(CC(=O)NCC(O)(COC)CO)C1 7097,N1(C(CCSCC)=O)CCCOC(CCNC(=O)Cn2ccc(C)n2)C1 7098,Cc1c(C(=O)NC2(CF)CCN(C(=O)C(F)(F)c3cscn3)C2)cnn1CCO 7099,C(=O)(C1=Cc2ccccc2C1)NC1(CNC(C(C(CC)O)C)=O)CC(F)(F)C1 7100,c1(OCC(=O)NCC(CNC(C(CC)C)=O)(C)O)cc(C(C)C)ccc1C 7101,CCC(C)(C)CC(=O)NCC(C1CCCN(C(=O)Cc2nnc(S)n2C)C1)(C)O 7102,c1(CC(=O)N(CC(C)CNC(C2CC2C2CC2C)=O)C)noc2ccccc12 7103,N1(C(CCOCCC)=O)CCC2CCCC12C(=O)NC(CO)C(C)(C)CO 7104,C1(C(N(C)CC2N(C(C(C3CCCC3)OCC)=O)CCC2)=O)CC(S(C)(=O)=O)C1 7105,S(=O)(=O)(c1ccn(-c2ccccc2)n1)Nc1c([N+](=O)[O-])scc1 7106,O=C(N=c1ccn(CCC(=O)N2CCCC2)[nH]1)c1ccnc(F)c1.C(CSCC)N 7107,C1(N(C(CN(C(=O)CCOC(C)C)CC)=O)C)CC2CCC1O2 7108,n1(CC(=O)N(C(CNC(CC2(OC)CCC2)=O)C)C)cnc(C(N)=O)n1 7109,C1(C(N(C(CNC(c2cncn2C)=O)C2CC2)C)=O)CCCN1C(=O)C(C)(C)C 7110,c1(C(N(C2CCN(C(C3CCC(=O)C3)=O)C2)CC)=O)cnn2cccc(Cl)c12 7111,c1(CC(N2CCC(F)(CNC(C(CCC#C)O)=O)C2)=O)ccc([N+](=O)[O-])cc1F 7112,c1(CC)nccnc1C(N1CC(OC)C(C(=O)NCCCCCO)C1)=O 7113,C1(C)(C(=O)NCC2CCN(C(C)C)C2)CCN(C(C23CC(CO2)C3)=O)C1 7114,CC(C)CC(C)C(=O)N1CCC(N(C)C(C2CC3C=CC2CC3)=O)CC1 7115,C(=O)(CC(=O)NC(C)C(=O)NCCCc1cscn1)OC 7116,Cc1nn2c(C(=O)NC3CN(C(c4cc(CF)on4)=O)CCC3C)c(C)nc2s1 7117,c1(C(=O)NC2CC3CN(C(C4N(C)C(=O)CC4)=O)C2C3)cc2c(nn1)CCCO2 7118,N1(c2n(CC(=C)C)c(C3CCSCC3)nn2)CC2C(C1)C2(F)F 7119,N1(C(CN(C(C)=O)C)=O)CCC2(CC(NC(C34CC(CCO3)C4)=O)CO2)C1 7120,C(C1=NOC(C)C1)NC(C(Cc1ccoc1)NC(CC(C)SC)=O)=O 7121,CCCCCC(O)CC(=O)NC(C1CCN(C(=O)C(C#N)CC)C1)C 7122,c1(C(C(=O)NCCSC)NC(=O)CN(C)C)cncn1C 7123,c1(C(=O)NC(CN(C(=O)CCc2cncn2C)CC)C)cc(N)cc(F)c1 7124,C1(C(=O)NCCN(C(c2ccc(NC(=O)NC(C)C)s2)=O)CC)CC2CC2C1 7125,c1(CN(C(C)C)CCN(CC(F)(F)C(F)F)C)cccc(C(=O)O)n1 7126,C1(C(N2CCCC(n3ccc(C(=O)OC)n3)C2)=O)CC2CC1CC2(C)O 7127,C1(CNC(CCCC#C)=O)CCN(C(=O)C(CCOC)OC)O1 7128,c1(C(C)O)ncc(C(=O)NCC2(CNC(c3ccc(CO)s3)=O)CCC2)s1 7129,C1(C(N(C(CNC(Cc2cnc(C)o2)=O)C)C)=O)Cc2cc(Br)ccc2O1 7130,C1(CNC(C(C)Cc2ccco2)=O)CN(C(c2ccc(F)s2)=O)CCO1 7131,C(c1ccco1)=CC(N1CCC1C(N1CCCC1c1ncc[nH]1)=O)=O 7132,c1(C(=O)NCC(CNC(c2c(C(C)C)nns2)=O)F)cccn(C2CC2)c1=O 7133,C(=O)(CC(CNC(C1C(C)(C)C1(F)F)=O)C1CCC1)N1CC(C(C)OC)C1 7134,c1(CNC(C(C2CC(NC(C3(C)CC3(F)F)=O)C2)F)=O)ccccc1O 7135,N1(C(c2c(CC)occ2)=O)CC(F)(F)CC1CNC(C1CC1C(=O)NCCO)=O 7136,Cc1nn(C)cc1NC(=O)CNC(=O)NC(c1ccccc1C(C)C)C 7137,Cc1c(C(=O)NC2CCN(C(=O)C=CCO)CC2CO)cc(C2CC2)n1C 7138,C(c1c(Cl)cccc1Cl)=C(C)C(=O)NC1CC(F)(CNC(C2CCOC2)=O)C1 7139,N1(CC(C)CN(C)C(=O)NCC2CC2c2ccc(N(C)C)cc2)CCCS1(=O)=O 7140,C=CC(CC)CC(=O)NC1CCCN(C(=O)Cc2csc(C3CC3)n2)C1 7141,C1(C(=O)NCC2(CC)CCCC2)(CC)CCCN1C(=O)C1CC1 7142,c1(C(N2CCCN(C(C(C)(C)OC)=O)CC2)=O)ccc2c(c1)C(=O)NCC2 7143,c1(OCC)ccc(Cl)nc1C(N1CC2C(C1)N2C(=O)CCC(=O)N1CCCC1)=O 7144,N1(C(C(C)OCC2CCCO2)=O)CC2CC1CN(C(=O)C(C)OCCc1nccs1)C2 7145,c1(C(=O)NC2(C)CCN(C(CC(C)C3CC3)=O)C2)ccc2c(c1)CCCCC2=O 7146,c1(C(N2CCC(F)(F)CC(C)C2)C(=O)NCCCOC)cccc2cnn(C)c12 7147,C1(C(=O)Nc2ccc(C)nc2)CCN(C(=O)C(O)C2CCC2)C12CC2 7148,c1(CC(=O)NCc2csc(C(N3CC4CC4C3)=O)n2)cccnc1F 7149,c1(OCC)cccc(C(N2CCCC(c3nn[nH]n3)(c3nn[nH]n3)C2)=O)c1CC 7150,C(=O)(C1=COCCO1)N(CCNC(c1cncc(OCC)c1)=O)CC1CC1 7151,c1(C(N(c2nccc(OCC)n2)CC2CCCN2)=O)ccc(F)nc1C 7152,CCCC(O)C(=O)N1CC(NC(c2conc2-c2ccc(Cl)cc2)=O)C(O)C1 7153,CCC(CC)(CO)C(=O)NCC(CC(F)(F)F)NC(C1CCCCC1C(N)=O)=O 7154,C1(NC(C2(OCC)CCOC2)=O)CCCCC1CNC(=O)CCC1CCOCC1 7155,c1(-c2cn(CC3N(C(C(CCC)N(C)C)=O)CCC3)nn2)ccc([N+](=O)[O-])o1 7156,CC(CN=c1[nH]cnc(Cl)c1Br)N(C)C(c1cnc2[nH]cncc1-2)=O 7157,N1(C(CCC2C(=O)NC(=O)N2)=O)CCCC2(CCN(C(c3cnsn3)=O)CC2)C1 7158,N1(C(C2CCCC(NC(Cn3c(C)ccn3)=O)CC2)=O)CCC2CCN(C)CC12 7159,CCCCC(CN=c1ccc(C(F)(F)F)n[nH]1)NC(C1(CCOC)CC1)=O 7160,C12(C(=O)NCCCC(C)(C)C)CCC(CN(C(c3cc(=N)[nH][nH]3)=O)C1)C2 7161,N1(C(c2scc(Cc3c(C)ncs3)c2)=O)CCCC1(C)c1cn(CCOC)nn1 7162,N1(C(c2nc(C)c(C)s2)=O)CCCCC12CC(NC(C1CC1C(F)F)=O)C2 7163,c1(C(N(CC(=O)NC(C)(C)C)C)=O)cc(F)c(Cl)c([N+](=O)[O-])c1Cl 7164,C1(C(C)C)CN(C(=O)C=CC(=O)NC2CC2)CCC1NC(=O)C(=O)N(C)C 7165,c1(-c2nc(NC(C3c4n(C)c(nn4)C3)=O)sc2)nc2ccc(C(F)(F)F)cc2s1 7166,c1(C(N2CC(CNC(C(CSC)O)=O)C(F)(F)C2)=O)cc(C)c(Cl)c(C)c1 7167,c1(OCCC)cccnc1C(=O)N(CCCCN(C)C(c1cccs1)=O)C 7168,C#Cc1ccc(C2(C(=O)NC(CNC(=O)CC3(OC)CC3)(CC)CC)CC2)cc1 7169,C#Cc1cnc(C(=O)NC(C2CCN(C(c3sccc3F)=O)C2)(C)C)c(C)c1 7170,N1(C(c2ccc(C)[nH]2)=O)CCCC(C)(CNC(C2(C)CCOC(C)C2)=O)C1 7171,Cn1ncc(C(=O)NCC2(C)CCCN2C(=O)CSc2n[nH]c(O)n2)c1C#N 7172,c1(CNC(C(=O)NC(c2ncccc2F)C)=O)ccc(OCCCN(C)C)cc1 7173,CCCCC(CNC(c1c(C)noc1C)=O)NC(c1cc(C(C)(C)C)n[nH]1)=O 7174,c1(CCC(=O)NCC2C3CN(C(C(=C(C)C4CC4)F)=O)CC32)cccc(Cl)c1Cl 7175,N1(C(c2ccsc2Br)C(=O)NCc2c(OC)cccc2)CCc2cc(Br)ccc21 7176,N1(C(CCOCCC)=O)C2CCC1CC(CNC(C1CCN(C)C(C)C1)=O)C2 7177,Cc1nn(C(C)C)c(C)c1CC(=O)NCCNC(c1cc(C(C)(C)C)no1)=O 7178,Nc1cccc(Cl)c1C(N1CCCC(N(C(=O)C#CC2CC2)CCF)C1)=O 7179,c1(C(=O)NC2(C)CCN(C(c3cncs3)=O)C2)cc([N+](=O)[O-])ccc1N 7180,N1(C(C(C(C)C)C2CCC2)=O)CCC(NC(=O)CCC2(C)CC2(F)F)C12CC2 7181,n1(CC(N2CC(C(N(CC(COC)O)C)=O)(SC)C2)=O)cccnc1=O 7182,C(=O)(C(C#N)C(C)(C)C)NC(CCC(=O)NC1CC(OCC)C1)C 7183,C(C(C)N=c1[nH]c2c(c(=NCC=CCl)[nH]1)COC2)Oc1cc(C)oc1C 7184,n1(C2CN(C(C(N3CCSCC3)C)=O)C2)cc(-c2ncccn2)nn1 7185,CCCCS(=O)(=O)N1CCCCC1C(N1CCCCC1COCC)=O 7186,CCC(C)(CO)C(=O)N1CCC(CN(C)C(c2cccc(C3CCCC3)c2)=O)C1 7187,C1(CC=C)(NC(=O)CCC2(C)CC2)CCN(C(=O)COC2CCCC2)C1 7188,c1(C(=O)NC(CC)(C)CNC(=O)C=Cc2cscn2)ccn2ncnc2c1 7189,C1(C(N(C2C(C)C2)C)=O)CCCCN(C(C2CCC2)=O)C1 7190,C1(C)(NC(C2C(C)CN(C)C2)=O)CCC(NC(C2C3CC4C(C3=O)C24)=O)CC1 7191,CCCCC(C)(F)C(=O)NC1CCC(C(=O)NCC(C)N(C)C)C1 7192,C1(NC(Cc2ccc(C)nc2)=O)CC12CCN(C(=O)C(C)S(N)(=O)=O)C2 7193,n1(CC(=O)N(C)C)cc(C2CN(C(C3CC(n4ccnn4)C3)=O)C2)nn1 7194,c1(C(=O)NCC(CCCC)NC(c2c(C)cnn2C)=O)nnc(Cl)cc1N 7195,C1(NC(=O)Cn2cnnc2O)COCCC1NC(c1ccn(C(F)F)n1)=O 7196,c1(SC)ccc(C)c(C(=O)NCC2COCCN(C(=O)Cc3cc(C)ns3)C2)c1 7197,c1(C(N)=O)ccnc(C(N2CC(OCCNC(=O)C(O)C3CC3)C2)=O)c1 7198,N1(C(C(C=CC)O)=O)CCCC(C2(NC(c3cc(=O)n(C)cn3)=O)CC2)C1 7199,N1(C(C2CCN2C(C2(n3cccn3)CC2)=O)=O)CCC(CO)C(O)C1 7200,C(C(=O)N1CCC(OC2CCOC2)CC1)(C(C)C)c1cnc(C)s1 7201,C(C(C)(C(=O)NCC(c1ccsc1)O)NC(=O)CCC(C)N(C)C)SC 7202,c1(OC)cc(NNC(=O)OC(c2c(C)n[nH]c2C)C)ncn1 7203,C1(CNC(N2CCC(c3ncn(C)n3)CC2)=O)CCc2nc(O)[nH]c2C1 7204,C(=O)(C1=NNC(=O)CC1)N1CC(NC(C2CCN(C(CC)=O)C2)=O)C(C(F)F)C1 7205,c1(C(=O)NC2CCCOC2)cn(CC2(C(N(C3CC3)CC)=O)CC2)nn1 7206,c1(NC(=O)NC2CCCN(c3ncc(CC)cn3)C2)c(Cl)ccnc1Br 7207,N1(C(C2CN(C(C(C=C=C)C)=O)CC23CC3)=O)CCc2ccccc2C1 7208,C1(CNC(c2c(C)[nH]cc2)=O)CN(C)CCN1C(=O)C(C)CC(C)C 7209,CC1(C)COCCC1CC(=O)NC1COCC1NC(=O)C(F)(F)c1cnccn1 7210,c1(CNC(C2CC(CNC(=O)CN3CC=CC3)C2)=O)ncc(F)cn1 7211,Cc1cc(CC(=O)NCc2cc(C(=O)NC(C)CC(C)O)cs2)on1 7212,c1(C(N(CC(C)NC(C2CCCN(CC)C2)=O)CC)=O)cc(C)nc(O)c1 7213,C1(c2n(CC=C)nnn2)(Nc2cc(C)c(C)c(Br)c2C)CCCN2CCSCC12 7214,C1(C(=O)NCCCN(C(C2C(=C)C2)=O)C2CC2)CCc2nc[nH]c2C1 7215,C1(CNC(C(C)(C)O)=O)CN(C(C2CCN(C3COC3)C2)=O)CCCO1 7216,N1(C(C2C(=C)CC2)=O)CCC(C(C)(C)CNC(=O)Cc2cccnc2OC)CC1 7217,c1(NCc2nc(C(=O)NCC)cs2)cccc(NC)c1.C(N)(=O)N 7218,N1(c2ccnc(-c3ccc(C)cn3)n2)CCOC(CO)CC1.N12CCC(CC1)C2 7219,C(=O)(CC(C)CCC=C(C)C)NCC1C2CN(C(C3(COCC)CC3)=O)CC21 7220,C1(CNC(c2n(C)nc(C(F)F)c2)=O)CC2CCC1N2C(=O)CN1CC2CC2C1 7221,N1(C(CC2C(C)CCN(C(C3OCCC3(C)C)=O)C2)=O)CCn2ncc(O)c2C1 7222,C1(C(N(CCC)CCC)=O)CC12CCN(C(=O)C(C)n1ccnn1)CC2 7223,N1(C(c2cncc(C)n2)=O)CCC2(C1)c1[nH]cnc1CCN2C(c1cnco1)=O 7224,Cc1ccc(CNCC2CCN(C(C3CNC(=O)N3C)=O)C2)cn1 7225,c1(CC(C(=O)OC)NCC(=O)NCc2ccc(C)c(C)c2)csc2ccc(C)cc12 7226,C1(NC(C(C)n2ccnc2)=O)CN(C(=O)COC2(C)CCOCC2)CC1C1CC1 7227,N1(C(c2ccc(OC)o2)=O)CC(C2CC2C(=O)NCCc2nncs2)C1 7228,c1(CNC(=O)Cc2cccc(F)c2)ccnc(OC2CCOC2)c1 7229,C1(NC(C2(C(C)C)COC2)=O)CN(C(=O)C(O)c2cnc[nH]2)CC1(C)C 7230,N1(C(C(C)=CCC)=O)CC(NC(c2c(C)noc2CC)=O)CC12CCCCC2 7231,C1(C)(C(N(CC(C)(C)NC(=O)CSC(C)(C)C)C)=O)CC(C#N)C1 7232,c1(C(=O)NC2C(CNC(=O)CCCCC(F)F)CCC2)cnc2cccnc2c1 7233,N1(C(C(CCSC)(C)C)=O)CCC2CCN(C(=O)Cc3ncc(C)o3)CC2C1 7234,CC1CCCCC1C(=O)NC(C1CN(C(c2cncnc2)=O)CCO1)C 7235,N1(C(c2n(C)nnc2)=O)CCC(=CCNC(=O)CC2CCCSC2)CC1 7236,N1(C(C(C)CNC(=O)CCCN(C)C)=O)CCCC(O)CC1 7237,c1(C(N2CCC(NCc3cccc(OC)n3)C2)=O)cc2sccc2[nH]1 7238,Cc1ccc2ncccc2c1NC(C1CCN1C(c1cccc(C(F)F)c1O)=O)=O 7239,C1(NC(C2CN(CC(C)C)C(=O)C2)=O)CCN(c2ncccn2)C(C)C1 7240,C1(CNC(c2c(C)coc2)=O)CCN(C(=O)CSCC(F)(F)F)CC1C 7241,N1(C(C(CC)(C)O)=O)CC2OCCN(C(c3cc(C)cc(C)c3C)=O)C2C1 7242,N1(C(c2c(C)n(CCC(C)C)nc2)=O)CCN(C(C2C=CCCC2)=O)C(CF)C1 7243,C1(C(N(CC(C)NC(c2c(N)ccc(CC)c2)=O)C)=O)CC2CC(O)CC(C1)C2 7244,CC#CCCCC(=O)N(C1CCCC(NC(c2nccc(F)c2Cl)=O)C1)C 7245,c1(OC)cccc2c(C(=O)NC3CCCCN(C(C4CNC(=O)N4)=O)C3)csc12 7246,C1(NC(c2c(C)nc[nH]2)=O)CC(CNC(c2nc(Br)c[nH]2)=O)C1(C)C 7247,c1(SCC)cnc(O)c(C(=O)NCCC(C)N(C(=O)C(C)N(C)C)C)c1 7248,C=C(C)CC(C(=O)N1CCCC1C(N1CCC(n2cnnn2)C1)=O)OC 7249,C1(C(N2C(CCCNC(C=NOC)=O)CCCC2)=O)CCC=CCCC1 7250,C(=O)(C(C)(O)CC(F)(F)F)N(C(c1ccc(Br)cn1)C)C 7251,C12(Cn3cc(CN4CCC(c5cn(C)nc5)CC4)nn3)CC=CCN1CCC2 7252,O=C(NN1CCCCC1)NCCOCCC1CCCC1 7253,c1(OC)nc(N2CC(C(C)NC(c3snnc3C(C)C)=O)C2)cc(C)n1 7254,N1(C(c2c(C)c(C#N)[nH]c2)=O)CCOC2CN(C(=O)CC(C)C(C)(C)C)CC12 7255,CCC(C)C(C(=O)NCCC1CC(NC(C2(C)CC(F)C2)=O)C1)NC(C)=O 7256,c12nc(C)c(o1)CNC(=O)C(c1ccccc1)NC2=O.C1(CC)CCCC2CC12 7257,c1(C(=O)NC2C(CNC(COCC=C)=O)COC2)oc2ccccc2c(=O)c1C 7258,c1(OC)ccc2c(=NCCC#N)[nH]c(N3CCC(Cn4cccn4)C3)nc2c1 7259,CC1CC(NC(c2ccnc(C3CC3)n2)=O)CN1C(c1cnn(C)c1Br)=O 7260,CC1(C)CCCOC1CNC(=O)CC12CCC1CN(C(=O)CC(F)(F)F)C2 7261,c1(C(C(=O)NCCOC)N(C)C)cnc(CC)s1.C12CCN(C1)CC(O)COC2 7262,C1(CNC(C(CC)OCC)=O)(CO)CCN(C(c2csc(SC)n2)=O)CC1 7263,c1(C(=O)NCC#CCNC(CC(C)O)=O)cc(Br)ccc1Cl 7264,Cc1ccc(N)c(C(=O)NC2CCCC(NC(=O)CC3CCCC4(CC4)C3)C2)c1 7265,c1(C(N2CC(C)N(C(=O)CCc3cc(Cl)no3)CC2)=O)cccc2oc(=N)[nH]c12 7266,N1(CC)CC2CN(C(=O)C=CCC3(NC(C4CC(=O)OC4(C)C)=O)CCC3)CC2C1 7267,c1(C(N2CC(NC(C(c3ccccc3F)(C)OC)=O)C2)=O)cnc(C(F)F)nc1 7268,C(CO)(C(C)(C)CO)NC(CCNC(C1(C)CC1(F)F)=O)=O 7269,C1(C(N(CCCN)CCO)=O)CCCN1C1CCC(c2ccccc2)C1 7270,c1cc(CCNCc2ccn3ncnc3c2)c2c(c1)CCCC2 7271,N1(C(C2CN(CCC)C(=O)C2)=O)CCCN(C(c2cncc(O)c2)=O)C(C)C1 7272,c1(N2Cc3c(C)cnn3CC2)nc(=NCC2CCO2)[nH]c2c1CCCCCC2 7273,C1(NC(C2C(C(=O)OC)C2)=O)CCC(NC(=O)Cc2ccccc2C)CC1 7274,C(C(=O)NC1CC2CCC1(NC(C1CCCCC1)=O)C2)(C(C)(C)C)NC(C)=O 7275,C(=O)(C(CCO)N(C)C)NCC(CC)NC(c1sc(C)nc1CC(C)C)=O 7276,C=CC1(C(=O)NCC(C2(O)CCN(C(=O)Cn3[nH]cnc3=N)C2)C)CCCCC1 7277,c1(C(=O)NCC(CNC(=O)C=Cc2ccc(C)nc2)OC)cc2ccccc2[nH]1 7278,C(=O)(C1CCCc2scnc21)NC1CCN(C(C2(CN(C)C)CC2)=O)CC1F 7279,C(=O)(C1=C(C)OCCS1)NC(COCC)C(=O)Nc1ccc(C)c(CC)c1 7280,C1(NC(C(C(C)C)OC)=O)CN(C(=O)CCc2ccc(F)nc2)CCC1C 7281,C1(Nc2onc(OC)c2Br)CCN(C(=O)CCCNC(=O)C(C)(C)C)CC1O 7282,c1(OC)ccc2[nH]c(C(N3CCC(NC(=O)C=C4CCC(C)C4)C3C)=O)cc2n1 7283,NS(=O)(=O)c1cc(C(=O)NCC2CCC(NC(=O)Cc3ccco3)C2)co1 7284,C1(C2(O)CCN(C(C3CCCC3S(C)(=O)=O)=O)CC2)(NC(C(CC)C)=O)CC1 7285,C=CC1(CC(=O)NCCC(C)NC(=O)C(O)Cc2ccccc2)CCCCC1 7286,CC(C)(C)C(CC(=O)N1CC(NC(c2ccc3c(c2)CCC=C3)=O)C1)C(F)F 7287,c1(C(N(C2CN(C(=O)Cc3csnn3)CC2F)C)=O)cc2cncn2c(O)n1 7288,Nc1cc(C(=O)NC(C2CCOC2)CNC(=O)C=C2CCSCC2)ccc1F 7289,N(C(=NCCN1CCOCC1)NCC1CN(C)CCN1C)CC(C)OC 7290,C1(C(NOCC#C)=O)(COC)C=CCN1C(=O)C(C)C1CC1 7291,C(C(C)(C)C(=O)NCC1(F)CCC(NC(C2(C)CC2)=O)C1)N(C)C 7292,CC1(C2(C(=O)NCc3cc[nH]c3C(N3CCC(O)(CN(C)C)C3)=O)CC2)CC1 7293,C1(NC(C2(C#N)CC2)=O)(CF)CCN(C(=O)Cc2ccccn2)C1 7294,C#CCC(C)(C)C(=O)NCCOC1CCN(C(=O)CC2CCOC(CC)C2)C1 7295,S(=O)(=O)(c1cc(C(F)(F)F)ccn1)N(CC(=O)Nc1ccccc1)C 7296,Cc1cccc2[nH]cc(C(N3CCC(C)(CNC(C45CSCC4C5)=O)CC3)=O)c12 7297,N1(C(C2CC(C)N2C(c2ccn(C)n2)=O)=O)CCc2cnccc2C1 7298,C1(C(=O)NCC(=O)OCC)CCC(NC(=O)C(F)C(=O)OCC)CC1 7299,Cc1ccc(-c2c[nH]nc2C(=O)Nc2ncc(C(C)C)s2)cc1C 7300,C(=O)(C(=O)N=c1ccc(C#N)c[nH]1)OCC(C)OCCN 7301,c1(C(N(CCN(C)C(=O)OC(C)(C)C)C)=O)cnn(C(F)F)c1 7302,C(=O)(CS(=O)CCC(F)(F)F)NCC1(NC(c2cc(C#N)[nH]c2)=O)CCCC1 7303,c1(C(C(=O)NCCCSCC)N(CCCCC)C)cn(CCOC)nc1C 7304,c1(CC(=O)N(C)CCOCCC(=O)NC2CC2(Cl)Cl)ccc(C(F)(F)F)nc1 7305,S(=O)(=O)(c1cnc(NC(c2nccnc2C)C)c(Cl)c1)NCC=CCCC 7306,N1(C(CN(CC(C)C)C(c2cnn[nH]2)=O)=O)CC(C)C(F)(F)C1 7307,C(=O)(C(C)C(F)(F)F)NCCCCCNC(C(c1cccc(C)c1)F)=O 7308,C1(NC(C(c2cccnc2)OC)=O)COC2(C1)CN(C(c1csnn1)=O)C2 7309,n1(CCNC(N2CCCC(C(C(=O)OC)(C)C)C2)=O)nc(C)c([N+](=O)[O-])c1C 7310,Cc1ccc(C)c(CCC(=O)NCC2CCCN2C(=O)C(O)CC(C)C)c1 7311,Cc1cc(C)c(C(=O)NC(C2CCCC2)CNC(=O)CC2CCC(C)C2)c(C)c1 7312,Cc1cccc(Br)c1S(=O)(=O)NC(Cc1ccccc1)C(=O)O 7313,C1(C(=O)NC2(C)CN(C(CCN(C)CC)=O)C2)CCc2ncnn2C1 7314,N1(C(CSCC)=O)CCN(C(=O)CC2C(=O)NN=C2C)C(CS(C)(=O)=O)C1 7315,O=C(CC(CNC(C1CC(F)C(=O)N1)=O)C1CCC1)NOCC1CCCO1 7316,C1(CNC(c2coc(Cl)n2)=O)CN(C(=O)CNC(=O)C(F)(F)F)C2CCN1C2 7317,Cc1cc(NC(=O)C(C2CCN(C(=O)CC3CCCC3O)C2)C)cc(O)c1 7318,C(=O)(C(O)CC(F)(F)F)N1C(C(N2CCCC(CC=CC)C2)=O)CC(F)C1 7319,N1(C(c2c(C)nc(Br)cc2)=O)CCN(C(=O)CCc2ncc[nH]2)C2(CC2)C1 7320,N1(C(C2N(C)CCCC2)=O)CCN(C(c2cccnc2F)=O)CC1C(F)(F)F 7321,C12(NC(c3nnnn3CCc3ccccc3)C3(C)CSC3)CC1CS(=O)(=O)C2 7322,C1(=CCNC(c2ncsc2C2CC2)=O)CCN(C(C2C(CC)(COC)C2)=O)CC1 7323,C=CC(C)(CC)C(=O)NC(c1ccccc1F)CNC(=O)C=Cc1cnc[nH]1 7324,c1(C(=O)NCC(C(C)(C)C)NC(CN(C)CCO)=O)ncc(Cl)cc1Cl 7325,c1(C(=O)NC2COCC2C(N2CC3CC2C3)=O)ccc2cc[nH]c2c1 7326,N1(C(C(C)(C)OC(C)=O)=O)CC(CNC(=O)CN(C)C2CC2)C(C)(C)C1 7327,C(C)(C(C(=O)NCCc1cccnc1C)NC(=O)C(C)OCCOC)OC 7328,CC1CCC(C)N(C(=O)CC2CN(C(c3cn(CCO)nn3)=O)CCO2)C1 7329,C12(NC(=O)OC(C)(C)C)CCCN(Cc3c[nH]c(-c4ccccc4)c3)CC1C2 7330,Cc1cc(N)c(C(N2CC3=C(C2)CN(C(C2(C)CC(F)(F)C2)=O)C3)=O)cc1C 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7349,c1(CC)cc(C(=O)N(C(C)CNC(=O)CCCC2CCCO2)CC)ccc1F 7350,O=S(=O)(c1ccc(NC2CCCC2CO)cc1Cl)N1CCC(C2CCCCC2)C1 7351,C(=O)(C1=C(Cl)CCOC1)NCC(CC)(C)NC(c1cccc2sncc12)=O 7352,c1(OC)ccc2c(c1)NCCN(Cc1ccccc1OC1CC1(F)F)C2 7353,N(C1CCCc2cc(F)ccc21)C(Cc1ccc(CN)nc1)=O 7354,CC1(C)C2CC(C(=O)NCC#CCNC(C3(F)CCCOC3)=O)CC12 7355,N1(C(C2C(CNC(Cn3c(=N)nc[nH]3)=O)CC2)=O)CC2CCCC2C12CC2 7356,N1(C(C(CC)OC)=O)CCN(C(C2(C#N)CC2(C)C)=O)CC1C 7357,C(=O)(C(Cc1ccccc1)S(C)(=O)=O)N1C(CC(=O)NC)CCCC1 7358,C1(C(=O)NC(C(C)C)(C)CNC(=O)C(O)Cn2cncn2)SC2C=CC1CC2 7359,Cc1ccc2ncc(C#N)c(N3CCN(C4CC4)C(C)C3)c2c1 7360,CCS(=O)c1ccccc1C(=O)NC1CN(C(c2cncnc2)=O)CC1C1CC1 7361,C1(CC)CN(C(=O)CO[Si](C)(C)C)CCN1C(=O)CC1CCC1 7362,CCCCC(C)CCC(=O)NOCC(=O)NC1CCN2CCC1C2 7363,c1(C(=O)NCCC(C)NC(C(CC)CC2CCCC2)=O)cc(OC)cc(C)c1 7364,N1(C(C(C)OCC(F)(F)F)=O)CCC(NC(=O)CCCC(N)=O)C(O)C1 7365,c1(CN(C)C(=O)NC2(c3ccccc3)CC2C(F)(F)F)cnc2ccccn12 7366,C=CC(C)(C)CC(=O)N1CCCC1C1CCCN(C(=O)CCN(CC)CC)C1 7367,c1(C(C)(C)C)c[nH]cc1C(N1CCCC1CNC(c1c[nH]nc1C1CCC1)=O)=O 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7386,N1(c2cc(C)cc(C)c2)C(=S)NC(c2cccc(Br)c2)C2=C1C(C)CN(C)C2=O 7387,Cn1ccnc1C(F)(F)C(=O)NCCN(C(C1CC(C(F)(F)F)C1)=O)CC1CC1 7388,N1(C(c2c(CC)noc2)=O)CC(C)(C)CCC1CNC(C1CC(S(C)(=O)=O)C1)=O 7389,C(=O)(C1=CCCN(C(c2cc(O)c(O)c(O)c2)=O)C1)NC(CCC)C 7390,C1(NC(C2(C)CC(F)(F)C2)=O)CCN(C(=O)CSC2CC2)C(C2CC2)C1 7391,c1(C(=O)NC(C)C(C)NC(=O)CCC2CCCCO2)ccc2cc[nH]c2n1 7392,N1(C(c2nc(=O)cc(N)[nH]2)=O)CCC2(CC1)CN(C(=O)CCc1cc(Cl)cs1)C2 7393,C1(CCNC(c2nocc2Cl)=O)CCCCN1C(c1ccsc1-n1cnnn1)=O 7394,C12(C(N(C(C)C(C)(C)O)C)=O)CC(CO1)N(C(C1CC3CCCC3C1)=O)C2 7395,C(CCCC(CO)NC(=O)CCc1cn(C)cn1)NC(C1OCCC(C)C1)=O 7396,C1(C(=O)NCCCC(=O)NC2CC2)CC2CC2N1C(=O)CC1NC(=O)NC1=O 7397,C1(C(=O)NCCC2(O)CN(C(CN(CCC#C)C)=O)C2)CC=C(C)CC1 7398,N1(C(C(CC#C)(C)NC(c2ccn(C)c(=O)c2)=O)=O)CCC2(COC(=O)N2)C1 7399,C(C(F)C(=O)NC(CNC(C1(CC2CCC2)CC1)=O)C1CCC1)N(C)CC 7400,N1(C(C=CC)=O)CCCC1(CNC(C1CN(CC)C(=O)N1)=O)COC 7401,CC1(C)CC(CC(N2CCCC2(C)CNC(c2coc(Cl)n2)=O)=O)CO1 7402,O=C(C1CCc2ccccc21)NCC1C2CC2CN1C(=O)Cn1ccnn1 7403,C(=O)(CC(CC)C(F)F)N1CCC(=CCNC(C(CC)C)=O)CC1 7404,c1(C(N2CCN(C(C3CC(CC)OCC3)=O)CC2C)=O)ccc2c(c1)CCCS2 7405,S(=O)(=O)(C1CC1)NCC(=O)NC(C1CCCN1C(c1nc(C2CC2)cs1)=O)C 7406,c1(N2CC=C(CNC(C(C)N(C)C)=O)CC2)nc2ncc(Cl)cc2o1 7407,Cc1c(-n2cc(C3CCN(C(=O)CC(C)C4CC4)C3)nn2)cccc1F 7408,c1(OCC(N)=O)cccc(C(=O)NC2CCC(NC(=O)CSC3CC3)C2)c1 7409,C1(C(=O)NC(CCC)CCCNC(C2(CC)CCC2)=O)CCc2nc(C)cn2C1 7410,Cc1ccc(N)cc1C(N1CCCC(F)(CNC(=O)CNC(=O)CC(C)C)C1)=O 7411,CCC(CC(C)C)C(=O)NC1(C)CC(C(=O)NC(C2CCCCC2)CO)C1 7412,CC1CSc2ccccc2CN1C(=O)Nc1ccc(C(N)=O)nc1O 7413,C1(NC(CC(C)c2ccncc2)=O)(CO)CCN(C(C2(CF)CCC2)=O)C1 7414,C(=O)(C(F)C(=O)N1CCC(NC(=O)CC=C(C)C)C1C(C)(C)C)OCC 7415,c1(NC(=O)CCCCBr)ccc(CNCc2ccc(F)nc2F)cc1F 7416,c1(N(C(C2CC2c2ccc(Cl)cc2)=O)CC2COC2)ccccc1Cl 7417,C(=O)(CCC(F)(F)F)NC1C(C)CN(C(=O)CCc2nnc(S)n2C)C1 7418,C(C(=O)Nc1ccccc1)(C(C)(C)C)N(C)Cc1ccc(C)cc1 7419,n1(CC)nc(C)c(CC(N2CC(NCc3cc(C)cnc3Cl)C(C)C2)=O)c1C 7420,C(=O)(C1CCCc2nc[nH]c21)N(CC(C)N(C(c1nc(OC)c(F)cn1)=O)C)C 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7475,c1(C(=O)NC2C(NC(C(C)(CO)NC(C)=O)=O)COCC2)ncc(Cl)cc1F 7476,CCC1=NOC(C(N2CCOCC2C(=O)NC(c2nc[nH]n2)C2CC2)=O)C1 7477,c1(C(c2n(CCCC)nnn2)NCC2(CO)COC2)ccc(F)cc1I 7478,CC1CCC(C(=O)N(C2CC3CC3C2)C)N(C(=O)Cc2ccon2)C1 7479,N1(C(C(C)(C)OCC)=O)CCC(C)(CNC(=O)CCc2cccc(F)c2F)CC1 7480,C1(F)(C(N(C)Cc2cnco2)=O)CN(C(=O)CC2CC(F)(F)C2)C1 7481,CC1(C)CN(C(c2coc(C3CC3)n2)=O)CCC1NC(=O)COCC1CCCO1 7482,C1(C(=O)NCC(C)(CO)NC(c2c(C)n(C(C)C)cc2)=O)CCCCC(C)(C)C1 7483,c1(SC)cccnc1C(=O)NCCC1CN(C(=O)CC2C(=O)NN=C2C)C1 7484,N1(C(COC2CN(C(c3cc(SC)oc3)=O)C2)=O)CC2CCCC2C1 7485,CP(C)(=O)C1(C(N2CC(O)(C3CCCN3C(=O)CC3CC3)C2)=O)CC1 7486,CC(C)(C)CC(F)C(=O)N1CCC(Cn2cc(C3(n4ccnn4)CC3)nn2)C1 7487,c1(OC(C)C(=O)NCC2CC(C)N(C(=O)CC(O)C3CCCC3)C2)ccc(F)nc1 7488,CC1(C)CCC(NC(N2CCC(OC(=O)NC3CC3)C2)=O)C(OCCCl)C1 7489,N1(c2nnc(COC)s2)CC2CC1CCC2NC(C1(O)CCSCC1)=O 7490,C1(C(N2C(CNC(C(CSC)C)=O)CCC2)=O)(NC(=O)OC(C)(C)C)CCCCC1 7491,C12(NC(C3C(CC)C3(F)F)=O)COC(C1)C(NC(c1cnn(C)n1)=O)C2 7492,c1(SC)cnccc1NC(C1CS(=O)(=O)N1)=O 7493,CC1CN(C(=O)COCc2cn(CC3CCO3)nn2)CC1(C)CC(=O)O 7494,N1(C(C2CC(=C)C2)=O)CCCC(C2CN(C(c3cc(O)n(C)n3)=O)C2)C1 7495,c1(C(N2CC(C(C)OC(C(=O)OC)OCC)C2)=O)ccc(C(=O)CC)cc1 7496,Cc1n[nH]c(C)c1C(=O)N(C)CC1(O)CN(C(=O)C(C)(C)C2CCOC2)C1 7497,CCC(C)(C)CN(C)C(=O)N(c1cccnn1)CCOC(F)(F)F 7498,C1(NCC(C)CC2CCC(F)(F)CC2)CCc2c(nnn2C)C1 7499,C(=O)(C1=CC2CCCC12)N(CC(CNC(c1cccc(SC)n1)=O)C)C 7500,Cc1nc(N2CCN(C(=O)COC3CC3(F)F)CC2)c2scc(C)c2n1 7501,CC1C2C(CCN2C(C2CCc3n[nH]cc3C2)=O)CN1C(=O)Cc1ccn(C)c1 7502,Cc1cc(C(=O)NCC(O)CN(C)C(C2OCC3CCCC23)=O)ccc1Cl 7503,N1(C(COCc2ncc(C)o2)=O)CCCC(C(N(c2ncncc2Cl)CO)=O)C1 7504,CC(C)C(C)(F)CNC(=O)CNC(=O)CNC(c1nc(Cl)cs1)=O 7505,c1(CN2C(C(=O)Nc3cc(OC)cc(C)c3)CSCC2)c(C)cc(O)cc1O 7506,CCC(CC)C(C(=O)NCC1(CNC(c2cnnn2CC)=O)CCOCC1)OC 7507,c1(C(C)C)[nH]nc(C(=O)NC(CNC(c2ccsc2)=O)CO)c1[N+](=O)[O-] 7508,C1(CCC(=O)NCC(C)=CC(=O)NCc2cccc(Cl)c2)CCCN(C)C1 7509,c1(N(C)C)cc(F)ccc1NC(=O)C(C)(C)NC(C1C2CC(=O)CC12)=O 7510,C12(CNC(C(C=C)OC)=O)CN(C(c3c[nH]nc3CC)=O)CC1CCO2 7511,N1(C(C2CCC3CCCCN23)=O)CCCCC1C1CCCN1Cc1cncs1 7512,C1(CNC(=O)C(O)C2CN(C(=O)COC3CCC3)C2)CCC(O)C1 7513,c1(C(N(CCC(C)NC(=O)Cc2cnn(C)c2)C)=O)ccc2nccnc2c1 7514,c1(C(N2CC3C(NC(CN(C)CC)=O)C(CC3)C2)=O)cc2c(cn1)OCCC2 7515,CC1=C(C(=O)NC2CN(C(c3ccc(C)nc3)=O)CCC2C(F)(F)F)CCO1 7516,C(=O)(C1CCc2c[nH]nc21)N1CCC(CC(=O)NCCC(C(=O)OC)(C)C)CC1 7517,C#CC1(C(=O)Nc2cnc(C3CC3)nc2)CCN(C(=O)CC=C(C)C)C1 7518,C1(C(=O)NC(c2n(CC)ccn2)C)COCCN(C(=O)CCc2ccnn2C)C1 7519,N1(C(c2c(CC)onc2)=O)CCOCC(NC(c2cc(C(C)C)ccc2N)=O)C1 7520,c1(CCC)c(C(N2CC3CC2C3NC(C2(OC(C)=O)CC2)=O)=O)nnn1CC 7521,C(=O)(CCCn1ccnc1)NCCCOCCC(=O)NC(c1cncnc1)C 7522,N1(C(CNS(CC)(=O)=O)=O)CCC(C2CC2NC(C2CC=CCC2)=O)CC1 7523,C1(C(=O)NC2C(NC(=O)CCc3ccnc(Cl)c3)C2)CN2CCCN1CC2 7524,C12(C(=O)NC(CNC(c3ccc(N)c(Cl)n3)=O)CO)CCCCC(=O)N1CCC2 7525,CCC(C)(CCNC(=O)CC1CC=CCN1C)NC(=O)CSC(F)F 7526,Cc1ccccc1C1(C(=O)NCC=CCNC(=O)C(F)n2ccnc2)CCC1 7527,N1(C(COCc2ccc(C)cc2)=O)CCC2CC(NC(=O)C=CCF)CCC2C1 7528,N1(C(c2c(Cl)sc(C)c2C)=O)CCC2(CC1)COC(CNC(c1cn[nH]c1)=O)C2 7529,C(CNC(C1CC12CCCC2)=O)(CC(=O)N1CCOC(CO)C1)OC 7530,C1(NC(CCc2ccc(C#C)cc2)=O)CCC(O)CN(C(=O)COCCOC)C1 7531,N1(C(C(=O)NC(C)CN(C)Cc2ccc(C3CCCO3)nn2)C)C(C)CCC1C 7532,C1(CNC(CCC=CC)=O)C2CN(C(c3nocc3C(C)(C)C)=O)CC12 7533,N1(C(CCC#C)=O)CCCC2(CCN(C(C3(S(C)(=O)=O)CCCCC3)=O)C2)C1 7534,C1(NC(CSCC=C)=O)CCN(C(=O)CSCCC(F)(F)F)C(C2CC2)C1 7535,c1(C(CC)=O)cc(C(=O)N(C2CC(NC(c3ncc(F)cn3)=O)C2)C)ccc1F 7536,N1(C(C2N(C(C(CC)(C)C)=O)C(C)C2)=O)CCC12CCCSC2 7537,Cc1cc(Cl)cc([N+](=O)[O-])c1C(=O)NC(C)CCNC(c1c[nH]nc1[N+](=O)[O-])=O 7538,CCCCS(=O)(=O)CC(=O)N1CC(C(C)Nc2cc(-n3ccnc3)ncn2)C1 7539,C1(CCCC)CCCCC1C(=O)NC1CN(C(=O)CCC(=O)OC(C)(C)C)C1 7540,C1(NC(c2c(SC)csc2)=O)CC2(C1)CC(NC(c1coc(C3CC3)n1)=O)C2 7541,O=C(CC1=CCCCC1)N1CC2CCCC1C2c1cn(Cc2cccs2)nn1 7542,Cc1ccc(NC(=O)CCC2CCC(NC(c3c[nH]c(C)c3)=O)C2)cc1CO 7543,C(CC1CCC1)(C(=O)N(C(C)C(=O)NCc1coc(C)n1)C)OC 7544,c1(OC)c(C(=O)NC2CC(O)CN(C(C3CCN(C)CC3)=O)C2)cc(F)cc1F 7545,c1(C(=O)NC(CC)(C)CNC(=O)C(C)CCCOC)c[nH]c2cc(C#N)ccc12 7546,C(=O)(CC(F)(F)C(F)F)NC(CCNC(c1cc(C)no1)=O)Cc1ccccc1 7547,C(=O)(C(CC(C)C)N(C)C)N(C1CCN(C(c2csc(C(C)C)n2)=O)C1)CC 7548,N1(C(c2n(C(C)C)ncc2)=O)CC2CCCC2(NC(=O)C(=O)NCC(F)(F)F)C1 7549,N1(C(C2CCCN(C(C)=O)C2)=O)CCCN(C(C2CCN2C)=O)CC1C 7550,C1(COC(C2ON=C(CC)C2)=O)CCCN(c2cnc(C#N)cn2)C1C 7551,N1(C(c2c(C)oc(C(C)C)c2)=O)CCN(C(=O)CC2(C)CCCO2)C(C(C)C)C1 7552,C1(C(=O)NCC(C(C)C)NC(=O)CC(C)(C)N(C)C)CCCC(F)C1 7553,c1(C(=O)NC2CN(C(C(CC)F)=O)C3(C2)CCC3)ccc2c(c1O)CCC2 7554,N1(C(C(C)NC(N)=O)=O)CCC(C(=O)NCc2nnc(O)o2)=C(F)C1 7555,C12(C(=O)NCCC3(NC(=O)C4=CSCCO4)CCC3)CCCC1CS(=O)(=O)C2 7556,C1(CNC(=O)NC2CCOC2)CCCN1C(c1cc(-c2ccccc2)[nH]n1)=O 7557,C1(C(n2cnc(C#N)n2)C)CCCC(C)(C)CC1.n12cc(nn1)CCCCC2 7558,N1(C(c2c(C)cc(F)s2)=O)CC(C)OC2(CCN(C(=O)CCc3ccon3)C2)C1 7559,c1(C(N2C3(CN(C(c4ccc(F)cn4)=O)C3)CC2)=O)cnc(O)n(C2CC2)c1=O 7560,C(CC(C(C)(C)C)NC(=O)CC1CC=CCC1)N(C)C(c1sccc1C1CC1)=O 7561,Cc1ccc(Cl)cc1CC(=O)NC1CC(n2cc(CC(C)CS(C)(=O)=O)nn2)C1 7562,C1(C(N(CC(C)N(C(C)=O)C)C)=O)CCN(C(=O)C(C)Cn2ccnc2)C1 7563,N1(C(CC(C)(C)c2cn(C3CCC(N(C)C)CC3)nn2)=O)CC2C(C1)C2(F)F 7564,C1(NC(c2cc(C(=O)OC)ncc2)=O)CN(C(C2CC(C)=NO2)=O)CC(C)(C)C1 7565,c1(S)ccc(Cl)cc1F.n1(CCCCC)c(CCc2ccco2)nnc1S 7566,N1(C(c2c(OCCC)cccn2)=O)CC(NC(C2CC2CC)=O)CC2(CCC2)C1 7567,c1(C(=O)NCC2CCCC(CNC(C(C)N3CCC3)=O)C2)noc2c1CCCC2 7568,N1(C(C(C2CC2)SC)=O)CCCC(C)(C)C1CNC(C1CC(CC(N)=O)C1)=O 7569,N1(C(C(n2cc(Cn3c(C)ccc3C)nn2)C)=O)CCOC(C2CC2)CC1 7570,C(=O)(C(C)(C)S(C)(=O)=O)N1CC(CC(C)NC(c2ccc(S(C)=O)cc2)=O)C1 7571,C(C(=O)NCC1CCN1C(C)=O)(C(C)C)NC(=O)OCC.C12CC(C1)NC(=O)C2 7572,N1(C(C(C(C)C)OCC)=O)CCC2(CCC(NC(=O)C3=NOCC3)CC2)CC1 7573,CCC(C(=O)NC1CC(C(=O)Nc2ccc(CO)c(F)c2)=CC1O)C(F)(F)F 7574,Cc1nn(C)c(NC2CC(C)CC(C)C2)c1C#N 7575,N1(C(c2ccc(COC)o2)=O)CC(CC(=O)NCCN(C)C(C)C)CC1(C)C 7576,N1(C(c2ccc(Cl)s2)=O)CCN(C(=O)C=CC2CCCO2)C(CO)C1 7577,CCC(C)(CN(C)N1CC(O)CC1CO)Oc1ccccc1 7578,c1(C(=O)NCC2CN(C(CS(CC)(=O)=O)=O)CC2C)cnc2c(C)cnn2c1 7579,C1(CCN(C)C)(CN2CCC(C(C(N3CCC(C)C3)=O)F)C2)CCOCC1 7580,C12(C(N3CCCC(C)(COC)C3)=O)CCCC1CN(C(=O)C(F)(F)CC)C2 7581,C1(NC(CCSCCC)=O)C=CC(C(=O)NC(C)Cc2cnccn2)C1 7582,C1(NC(C2(C)ON=C(C)C2)=O)CN(C(=O)C(C2(O)CCCC2)F)CC1(C)C 7583,Cc1ccc2c(c1)C(C(=O)NCC(F)CNC(c1ncccc1CO)=O)OCC2 7584,N1(C(CSCCC)=O)CCCC1C(C)NC(=O)C(C)OC1CCOC1 7585,CC1CCC(NC(=O)C(O)C2CCC2)CN1C(=O)CCCC1CC1 7586,N1(C(c2ccc(SC)o2)=O)CC(NC(=O)CCc2ccc(O)nn2)C(C)(C)C1 7587,C1(C#N)(C(=O)NCCC(C)N(C)C(c2cc(-c3cccs3)on2)=O)CCSCC1 7588,N1(C(Cn2ncn(C)c2=O)=O)CCC2CC1CN(C(=O)CCC1CC1(C)C)C2 7589,C1(NC(CN(C(=O)C(CSC)OC)CCC)=O)CCN(CCOC)C1 7590,c1(N(CCC)C)ccc(C(N2CC(CC(=O)O)C(O)C2)=O)cc1 7591,c1(C(=O)NCCN(C(C(Cc2c(C)noc2C)C)=O)C)ccc(C#N)nc1 7592,N1(C(C2(CC)CCCC2)=O)CCN(C(=O)COCCSC)C(C2CC2)C1 7593,c1(SCC(=O)NCCC(C)N(C)C(C2COC3(CCC3)C2)=O)ccsc1[N+](=O)[O-] 7594,S(=O)(=O)(c1cnn2ccc(=NCC3(Br)CC3)[nH]c12)N1C2CC(CC)CC1CCC2 7595,C12(NC(C3CCNC3=O)=O)CCCC1N(C(=O)COc1ccsn1)CC2 7596,N1(C(CC(=O)N(C)C)=O)CC(NC(c2cccc(CS(C)=O)c2)=O)C2(CCC2)C1 7597,c1(C(=O)NC2CCN(C(CCC#CC)=O)CCC2CO)cc2c(Cl)ccnc2s1 7598,C12(c3c[nH]nn3)COC(C1)C(O)C2.N1(C(CC2CC(CC)C2)=O)CCCC1C1CC1 7599,C1(O)(C(C(=O)N(C2CCOC2=O)C)F)CN(C(=O)C=CC(=O)NC2CC2)C1 7600,C1(C(=O)NC2C(CNC(c3ncc(C)c(C)c3)=O)CC2)CC(C)CC(C)(C)C1 7601,n1(CC)ncc2c1CCCC2NC(=O)NC(c1ccccc1)(C)C 7602,C(=O)(C(C)S(C)(=O)=O)N(C1CCN(c2cc(C)ncn2)CC1)CC1CCCO1 7603,C1(S(C)(=O)=O)(C(=O)NC2C(CNC(c3[nH]cc(CC)c3)=O)C2)CCCC1 7604,C12(CC)CC(C(=O)NCC(C)(CO)NC(=O)Cc3cn[nH]c3)(CO1)C2 7605,c1(C(=O)NCCN(C(=O)C(C2CCCCCC2)O)CC)cc(C)cc(Cl)n1 7606,N1(CC)N=C(C(=O)N2CCCC(C)C2CCNC(=O)COC(F)F)CCC1=O 7607,C1(CC(=O)NC2CCC(N(C(C(CC)N(C)C)=O)C)CC2)C(=O)N(C)N=C1C 7608,N(C(=NC1CCS(=O)(=O)C1)N1CCC2(CC1)CC(O)c1nn(C)cc1O2)C(C)C 7609,N1(C(c2cnc(C)nc2)=O)CC(NC(=O)C=Cc2cc[nH]c2)C2(CC2)C1 7610,N1(C(C(c2cn(-c3c(C)c(F)ccc3)nn2)C)=O)CCCc2sc(C(=O)O)cc2C1 7611,c1(C(N2CC(COC)(CNC(=O)C(C)C3CCC3)C2)=O)cccc(CC#N)c1 7612,c1(CNC2C(C(=O)NCc3c(C)cc(Br)cn3)CCCC2)cc2ccncc2[nH]1 7613,CCC(C(=O)NC1CCN(C(c2cc(O)nc(O)n2)=O)C12CC2)C(F)(F)F 7614,N1(C(CCC=C=C)=O)CCC2CN(C(=O)CN3C(=O)C(=O)N(C)C3=O)C2C1 7615,C(=O)(C(CNC(=O)CC(O)C1CCCC1)C(C)(C)C)NCCC=CCCC 7616,C(=O)(C1=CCCN(C(=O)CC(F)(F)F)C1)N(CC(N)=O)C 7617,Cc1ccc(C(N2CCC(CN(c3ncnc(Cl)c3F)C)C2)=O)cc1C 7618,CCN=c1[nH]c(COC(=O)N(C2CC(O)C2(C)C)CC)cs1 7619,Cc1cccc(C(=O)NC2CC(NC(C3(NC4(F)CC4)CC3)=O)C(O)C2)c1 7620,N1(C(c2ccnc(C)n2)=O)CC2CC(NC(c3ccc(C)c(F)n3)=O)C2C1 7621,C(=O)(C(CC)CC(F)F)NC1(CN(C(c2cc(CC)c(F)cc2)=O)C)CC1 7622,Cc1cc(C(=O)NC2CC(NC(C3(Br)CC3)=O)C2)[nH]c1C 7623,N12CCC(OC)(CC1)CC2.c1(NC(C2(C)CC(=C)C2)=O)ncnc(O)c1Br 7624,c1(C(=O)NC(CC(C)NC2C(OC)CCCC2)C)c(C)cccc1[N+](=O)[O-] 7625,n1(CC(=O)NC(C2(CNC(C3OCCCO3)=O)CC2)C)cnc(Br)n1 7626,CC1(C)CCC(CNC2CN(C(=O)C(=O)N(C)C)C(C)(C)C2)OC1 7627,N1(C(C(n2cc(C)nc2)(C)C)=O)CCC2(CCC2)C(NC(C2CCCC2O)=O)C1 7628,c1(NC)ncccc1C(=O)NCCC1CC(NC(=O)CCC2CC2C(C)O)C1 7629,c1(OC(C)(C)C)cc[nH]c(=N)n1.c1(C(C)(C)OCOCC)cn(CC(=O)O)nn1 7630,CC1C(C)N(C(=O)CSC(C)(C)C)CCN1C(C1C2CCC1(c1ccco1)C2)=O 7631,c1(C(N2CCCC(CCNC(c3ncn(CC)n3)=O)C2)=O)cnc2cc[nH]c2c1 7632,C1(C(N2CC(CC(C)NC(c3n[nH]cc3-c3ccccc3)=O)C2)=O)CCC=CO1 7633,C(=O)(C(C(C)(C)C)c1ccccc1)N1CC(NC(CCCSC)=O)C(C)C1 7634,Cc1nc(N2CC(NC(=O)CCC(C)(C)[N+](=O)[O-])C(C)C2)c(Cl)cc1C#N 7635,c1(C(=O)NCC(C)(CNC(C2C=CCCC2)=O)OC)cn(C)nc1C(C)C 7636,CC1C(NC(=O)CCc2cn[nH]c2)CCN1C(=O)CN1CCOCC1=O 7637,C(C1CCOCC1)=CC(=O)NCCC1CS(=O)(=O)C1 7638,CCCC(O)CCNC(=O)CSC.C1(=O)CCOCCN1C 7639,Cn1ccc(=O)c(C(N2CCC(O)(CNC(=O)C(F)n3cccn3)CC2)=O)c1 7640,c1(CC(=O)NC2CN(C(c3cn(Cc4onc(C)n4)nc3)=O)C2)cccc(F)c1 7641,N1(CC(=O)N(c2nccs2)CC(N2CCCC2)=O)CCc2cccc(F)c21 7642,C1(C(C)C(=O)NCCn2cnnn2)CCCN(C(C2SCCS2)=O)C1 7643,c1(C(=O)OC)cc2c(cc1NCCc1ccc(C)cc1Cl)CN(C(=O)OC)CC2 7644,c1(OC)cc(Br)cc(CN2CCCC2(C)C(=O)Nc2cnc3cc[nH]c3c2)c1O 7645,C=C(Cl)CC(C(=O)NCC(C)(C)C1CC1)NC(C1CC(=O)OC1(C)C)=O 7646,c1(CC)noc(C(N2CCSCC2CCNC(c2cnc(C)nc2)=O)=O)c1C 7647,N1(C(C2CN(C(c3c(C)ccc(OC)c3)=O)C2)=O)CCC2(CC1)CC2(F)F 7648,c1(C(N2CCCOC(CCS)C2)=O)cnc2c(Br)n[nH]c2c1 7649,c1(N2CCCC(C(C)NC(CCOCC#C)=O)C2)cc(-c2ccco2)nc(C)n1 7650,Cn1cnc(I)c1C(c1nnnn1CC(F)F)NC1(C2CCCO2)CC1 7651,C(=O)(CC(F)(F)C(F)(F)F)NC1CCCN(C(C(C)CC2CCCCC2)=O)C1C 7652,C1(NC(C(CC)Cc2ccccc2)=O)C(C)CCN(c2cncc(Cl)n2)C1C 7653,c1(CC(N2CC(NC(c3ccc(Cl)nc3Cl)=O)C(F)C2)=O)cc(F)c(F)cc1Br 7654,C1(NC(C(C=C)(C)C)=O)CC2CC(CNC(=O)CN(C)S(=O)(=O)N(C)C)CC2C1 7655,C1(NC(C(=O)NCC)=O)CCSC12CN(C(=O)C(C(C)C)NC=O)C2 7656,c1(OC)ccc(F)c(CC(N2CCOCC2CNC(C2CCNC(=O)C2)=O)=O)c1 7657,n1(CC(=O)OCC)nc(-c2cccc(F)c2)nc1-c1c[nH]c(=O)cn1 7658,c1(C(=O)NCC=CCNC(C2C(C=C(C)C)C2(C)C)=O)cc(N)c(Cl)c(O)c1 7659,c1(C(=O)NCC2(C(C)(C)O)CN(C(=O)CC3CCCC3)C2)cn2cccnc2n1 7660,C(CC(=O)NCC1CC(NC(=O)C(C)n2ccnc2)C1)OCCCOC 7661,CC1(C)CCC(C(=O)NCCC2CCCN2C(c2cc(O)cs2)=O)C1 7662,c1(OC)ccc(C(=O)NCC2CC2NC(=O)C(C(C)C)OC)c(OC)n1 7663,Cc1ccc(C(N2CC3(C2)CN(C(=O)C(=O)N(C)C)CC3CO)=O)c(N=[N+]=[N-])c1 7664,c1(OC)cncc(C(=O)N(C(C)CNC(=O)CC2CCC(=O)O2)C)c1C 7665,Cc1c(C(N2CC3CC2CN(C(=O)C=CC2CC2)C3)=O)nn2ccccc12 7666,CCCCCC(F)C(=O)N1CCC(C)C1C(=O)NCCc1nc[nH]n1 7667,c1(N(CCC)C)ccc(C(N2CC(CC(C)NC(=O)C(F)C(C)C)C2)=O)cc1 7668,C1(NC(CCC(=C)C)=O)CCC2(CC1)CN(C(=O)C1=COCCO1)CCO2 7669,c1(C(=O)NC(CN(C(=O)CCC2CC3CCC2C3)C)(C)C)sc([N+](=O)[O-])cc1Cl 7670,c1(-c2nc(CC(CC)C)nn2C(C)C(F)(F)F)cc2nccnc2cc1C 7671,CC(C)CS(=O)(=O)CCC(=O)NC1COC2CN(C(C3(C)CNC(=O)C3)=O)CC12 7672,c1(C(=O)NC2(CN(C(CCC(C)OC)=O)C)CC2)ccc(Cl)c(C)c1 7673,N(C1CCCc2c(Br)cccc21)C(c1n(CCC)nnn1)(C)C1CC1 7674,N1(C(CC2(NC(c3cccc(C(C)C)c3)=O)CCC2)=O)CCC(O)C(C)(CO)C1 7675,C1(CC)CCN(C(c2ccc(=N)[nH]c2)=O)C(C(=O)NC(C)CCCO)C1 7676,CC(C)CC(O)C(C)C(=O)NC(Cc1ccco1)C(=O)NCCCC(C)CO 7677,C1(NC(c2c(CCC(=O)OC)cccc2)=O)CN(C(=O)CC2CC2)CCC1(C)C 7678,C(N=c1cc(C(F)F)nc[nH]1)C1(NC(=O)CCCc2cccs2)CCOCC1 7679,N1(C(=O)Cc2ccc(Cl)s2)CCC(O)(C(N2CCC(CN3CCCC3)CC2)=O)C1 7680,C(=O)(C1CCCc2nn(C)cc21)NCCC(C)(C)NC(CC(C)NC(N)=O)=O 7681,C1(C(=O)NC2(CCOC)CCN(C(=O)Cn3cncn3)C2)C2CCC(C2)C1(C)C 7682,N1(C(c2ccc(C#C)cc2)=O)CCCC2CN(C(=O)C(n3ccnc3C)C)CC12 7683,N1C2CCC1CC(=O)NC2.c1(CC)cc(Cc2cn(CC3CC3)nn2)cc(CC)c1 7684,c1(N2CCC=C(C(=O)OC)C2)ncnc2c1ncn2C1CCC(O)(CO)CC1 7685,N1(C(c2c(CC)occ2C)=O)CC(NC(=O)CP(C)(C)=O)CC(O)C1 7686,C=CCCCC(C)(C)C(=O)NC1CCOCC1NC(=O)C(c1ccnn1C)O 7687,Cc1cc2[nH]c(C(N3CC4CC3CC4CNC(C3CCC(C)O3)=O)=O)cc2s1 7688,Cc1c(C(N2C3CCC2CN(C(=O)C(O)C(C)C)C3)=O)sc2ccnc(O)c12 7689,CCC(CN(C)C)CC(=O)NC(C(=O)N(C1CCSCC1)C)C1(O)CCC1 7690,c1(CC(=O)N(CCCN(C)C(C2CC2(F)F)=O)C)ncccc1Br 7691,C1(NC(C2CC23CCC3)=O)COCCC1NC(C1CCS(=O)CC1)=O 7692,N1(C(c2cc(C)n(C)c2)=O)CC(NC(c2ccccc2C#N)=O)C2(CCC2)C1 7693,C(C1CCOC1)=CC(=O)NC(C(=O)NCC1CC12CCC2)C1CCCC1 7694,Cc1cc(F)sc1C(=O)NCC(O)CC(=O)N1CCC(c2ncco2)C1 7695,c1(C(=O)NC(CNC(C(C2CCC2)OC)=O)C)cc(O)c2cnn(C)c2c1 7696,N1(C(C(C)NC(COC)=O)=O)CCCCC1C(N1CC2CC2(CO)C1)=O 7697,CCC(CC(=O)NCC1CCCCCN1C(=O)COCc1nnc(C)s1)C(C)C 7698,c1(CC(=O)NC(C)CCS(C)=O)ccc(Br)c(C#N)c1 7699,C(=O)(CC(CC#C)c1ccccc1)N1CCCC(N(C(C(F)=CC)=O)CCOC)C1 7700,C1(CN(C(=O)CC2CCOCC2)CC)CCN(C(c2cnn(CC)c2)=O)CC1 7701,C1(CNC(c2cc[nH]n2)=O)(NC(c2ccc(-c3ccccc3)o2)=O)CCCCC1 7702,C1(NC(c2[nH]nnc2C2CC2)=O)CN(C(=O)Cc2cncc(F)c2)C2CC12 7703,c1(C(=O)NC(CC)CN(C)C(C2(CC)CCOCC2)=O)ncc(C)cc1Br 7704,C(C(C(C)(C)C)CC(=O)OC)NC(=O)NC1CC(OCC)C1 7705,C(=O)(C1(C)CCn2c(C)nnc21)NCC1CN(C(COCC)=O)CC(C)(C)C1 7706,Cc1cccc2[nH]c(=NC3CCC4CN(C(C5CC5F)=O)CC4C3)sc12 7707,CC1(C(F)F)CC1N(C(=O)CCOC(F)F)C1CC1 7708,c1(C(N2CCC(NC(C3(C=C)CC3)=O)C(C)C2)=O)ccc2c(c1)CC(=O)N2 7709,C1(NC(=O)NC2CCN(c3ncco3)C2)CC2OCCC12 7710,C1(CNC(c2cc(CCC)n(C)n2)=O)CCC(C)CN1C(=O)C(C=C)OC 7711,C(=O)(C(C)C(C)C)NCC1(F)CC(CNC(C2C(OC)(OC)CC2)=O)C1 7712,CC(C)S(=O)(=O)CC(=O)NCC(CNC(C1C2CCCCC12)=O)CO 7713,N1(C(CNC(c2c(CCC)n[nH]c2)=O)=O)CC2CC1CS2 7714,c1(C(N2CC(C)C(CCNC(=O)CSc3nncs3)C2)=O)ccccc1C#N 7715,C(=O)(C1=CC(C)(CC)C1)N(CC1CCN(C(CC(=C)C)=O)CC1)CC 7716,c1(C(N2CCC(NC(C(CC)C)=O)C(F)C2)=O)nn(C)c2ccc(Br)cc12 7717,c1(C(=O)NC2CCN(C(C3(OCC)CCOC3)=O)C2)cc(F)cc(C)c1N 7718,c1(C(=O)NCC=CCNC(=O)CC2CC(F)C2)ccccc1C#CC1CC1 7719,Cc1[nH]cc(C(=O)NC2CC(CO)N(C(=O)CCCN(C)C(C)C)C2)c(=O)c1Cl 7720,c1(OC)ccc2c(=NCC3CN(C(C)=O)C3)[nH]c(=NC(C)CS(C)=O)[nH]c2c1 7721,N1(C(CC=C)=O)CCCCC(C2CN(C(c3ccc(O)c(N)c3)=O)C2)C1 7722,C1(NC(CC(CC)C)=O)CCN(C(=O)C(C)NC(=O)CC(C)(C)C)C1(C)C 7723,N1(C(C(C(C)O)NC(C(CC#C)O)=O)=O)CCCCC1C#C 7724,c1(OCCCC)ccc(C(=O)NCC(CNC(=O)CCn2ccnc2)OC)cc1 7725,C1(NC(c2occ(C(=O)OC)c2)=O)CC2CCC1N2C(=O)CC1CCOC1(C)C 7726,C1(CCNC(CC(=O)N(C)C)=O)(NC(C2CC23CCCC3)=O)CCOCC1 7727,n1(CC(C)C)cccc(-c2nc(-c3cncc(F)c3)nn2C2CCCSC2)c1=O 7728,c1(C(N2CCC(CNC(c3c(C)nc(C)s3)=O)C2)=O)oc(P(C)(C)=O)cc1C 7729,c1(C(=O)OC)cncc(-c2cccnc2N2CCC(O)CC2)c1 7730,N1(C(CCC#C)=O)CC(C)C(NC(c2cnc(S(C)(=O)=O)s2)=O)C(C)C1 7731,c1(CN(C)C)cccc(C(=O)NCC=C2CCN(c3ncc(Br)cn3)CC2)c1 7732,C1(C(N(CCCCCNC(=O)Cc2nn(C)cc2Cl)C)=O)COCC(C)(C)O1 7733,C1(CC(C)C)(CNC(C2(C(N)=O)CCC2)=O)CCNC1=O 7734,CCC(C(F)C(=O)OC)NC(c1cccc(C(F)(F)F)c1)(C)C(=O)OC 7735,c1(C(N(CC(C)NC(C2CC(=O)N2)=O)C)=O)ccc(F)c(O)c1 7736,C#CCC(C)(C(=O)N(C1CCNC1=O)C)NC(=O)C(CCC)=CCC 7737,N1(C(C2CCCCCCN2C(=O)C#CC2CC2)=O)Cc2cccnc2C1 7738,c1(CC(=O)NCC(CNC(c2[nH]cc(CC)c2)=O)C)sc(CC(F)(F)F)nc1C 7739,c1(C(N2CC(CC=C)(NC(=O)Cc3ccc(O)nc3)C2)=O)ccc(Cl)c(C)c1O 7740,c1(N(CC(C)O)C(=O)NCc2cc(Cl)ccc2F)ccc2c(c1)OCCO2 7741,n1(C(C)C)cc(C(N2CC(C)(NC(=O)C(=O)NCC3CC3)C2)=O)c(O)nc1=O 7742,c1(C(N(CCCCN(C(CCCC(C)=O)=O)C)C)=O)[nH]c2c(c1C)CCCC2 7743,C1(O)(CNC(CCC2N(C)CCC2)=O)CCN(C(C2(C)CCCCO2)=O)C1 7744,Cc1cc(S(=O)(=O)NCCCc2cccc3c2OCCO3)cnc1C(F)(F)F 7745,c1(C(=O)OCC)ccnc(N(CCC(C)NC(C2(CC)CCC2)=O)C)c1[N+](=O)[O-] 7746,C=CCC(C)(CC)C(=O)NC(CNC(c1ccc(-c2cc[nH]n2)cc1)=O)CC 7747,c1(NC)ccc(F)cc1C(=O)NC1CCC(C)N(C(c2sccc2OC)=O)C1 7748,Cc1conc1C(=O)NCC1(CNC(C2CCC(=O)O2)=O)CCC1 7749,Cc1ccccc1C=CC(=O)NCC12CC1CN(C(=O)Cc1cnc(C)o1)C2 7750,c1(C(N2CCC(C(C)NC(c3c(C)nc(Br)s3)=O)CC2)=O)ccc(F)c(F)c1Cl 7751,C=CCC(CC(F)F)NC(C1C(CC)CCN1C(c1cccc(F)c1)=O)=O 7752,N1(C(C2(CC)CCC2)=O)CC2CCCC2(NC(=O)CCN2CCCCCC2)C1 7753,C1(OC)CC(CCNC(=O)CCc2cnn(C)c2)N(C(c2cnc(C)n2C)=O)C1 7754,C12(CNC(C(CC)(F)C(=O)OC)=O)CCCCC1N(C(C1CC(O)C1)=O)CCC2 7755,N1(C(C2C(C=C(C)C)C2(C)C)=O)CC(C)C(C)(C)C1.C(=O)(C1=CCCCO1)N 7756,C(=O)(C(CNC(=O)C(C)NC(N)=O)OC)N(CCCF)CC 7757,C(=O)(C1=CCCOC1)N(C(CC(=O)NCc1nc(CC)oc1)(C)C)C 7758,C1(C(N2C(CN(C(=O)CCc3ccoc3)C)CCC2)=O)CC(F)C(=O)N1 7759,N1(C(=O)CNc2ccccn2)CC(C(N2CC(N3CCNC3=O)C2)=O)C2(CC2)C1 7760,Cc1nc(-c2ccccn2)sc1C(=O)NCC1CN(C(C2CCCOCC2)=O)C1 7761,C1(C(=O)NCCC(C)NC(C2CNC(=O)CC2C)=O)CC2CCCCN2C1 7762,CC1(CC(=O)NC(CO)CCC2CC2)CCN(C(=O)CCCn2cccn2)C1 7763,C1(C(=O)NC(COC)C)CN(C(c2cnc(C(C)=O)cn2)=O)CCN1 7764,CC1CC2CN(C(=O)C=CC(=O)OC(C)(C)C)CC2N1C(C1CNC(=O)N1)=O 7765,C1(CNC(Cc2ccc(C)cc2)=O)CC(C(=O)NC(c2scnc2C)C)=NO1 7766,C#CCCC(C(=O)N1CCCC(O)(CC)C1)NC(=O)CCCC1CC1 7767,c1(CC(=O)NC2CC(O)CN(C(=O)CC3CC3)C2)c[nH]c2ncccc12 7768,C(=O)(C(C(C)(C)C)SC)NC(CN(C(c1cnc(Cl)s1)=O)CC)C 7769,Cc1c(C(=O)NC(CNC(C2CCCN2C(N)=O)=O)CO)oc2ccc(Cl)cc12 7770,N1(C(C=CC(C)C)=O)CC2CCN(C(c3ccncc3C(F)F)=O)CC12 7771,N1(C(C(C)(F)F)=O)CC2(CCCN(C(=O)C=Cc3ccc(C(F)(F)F)cc3)C2)C1 7772,c1(N(C(C(=O)NC(COCC)C(C)C)=O)C)cc(Br)cn1C 7773,CC(C)CC(CNC(c1cncc(C2CC2)c1)=O)NC(=O)C(C)c1ccco1 7774,c1(CC)cn2c(n1)CC(C(N1CCCCC1CNC(=O)CCc1cnoc1)=O)C2 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7880,c1(C(=O)NC(CCC)CNC(=O)C(C)NC(=O)NC)ccsc1C#N 7881,N1(C(CC2(OC)CCC2)=O)C2CCCC1CN(C(C1CC(O)C1)=O)C2 7882,n1(C(CC)CC)nccc1C(=O)N(CC(C)(C)NC(=O)C(CO)N(C)C)C 7883,c1(C(N2CC(C(N3C(COC)CCC3)=O)C(O)CC2)=O)n[nH]c2c1CCC2C 7884,C1(C(=O)NCCN(CC(C)O)C(c2cc3sccc3s2)=O)CCC(C)(C)CO1 7885,c1(C(C)(F)F)cccc(C(=O)NC2CN(C(C3CCCC3CF)=O)CC2O)n1 7886,c1(C(NNCC=C)=O)sc2cc(Cl)ccc2c1Cl 7887,C=CCC(C)C(=O)NCC(C(=O)NCc1ncoc1COC)N(C)C 7888,Cc1c(F)ccc(C(=O)NCCCC2CN(C(c3ccc[nH]3)=O)CCO2)c1Cl 7889,N1(C(COC)=O)CCN(C(=O)CP(C)(C)=O)C(CO)C1 7890,Cc1cc2[nH]c(C(=O)NC3CC4CC3N(C(c3ccsc3)=O)C4)cc2o1 7891,N1(C(c2nc(NC(C)=O)sc2)=O)C2CCC1C(NC(=O)CC1CC3CCC1CC3)C2 7892,C(CCN=c1ccc(C(F)(F)F)c[nH]1)N(C)C(c1cccc(Br)c1Br)=O 7893,Cc1nc(N2CCC(F)C(NC(=O)OC(C)(C)C)C2)c(C)c(C)n1 7894,N1(C(c2cc(C)[nH]n2)=O)CC(C)OC2(CCN(C(=O)Cc3cccn3C)C2)C1 7895,c1(NCC(C)(CC(C)C)NC(CCCCCCC)=O)ncnc2c1nnn2C 7896,C1(C(C)(CSC)NCCCOCCO)CCOCC1 7897,CC(CN(C)C)CCC(=O)N1CC(CNC(c2cccs2)=O)CC1(C)C 7898,N1(C(CC2C(C)CCN(C(CC=CCC)=O)C2)=O)CC(C)(CO)CC1(C)C 7899,C1(CNC(=O)Cc2cccc(F)c2)CN(C(C2CCCC(F)(F)C2)=O)CC12CC2 7900,N1(C(CN(CC)CC)=O)CC2CCC1C1CN(Cc3ccccc3)CC21 7901,C1(NC(c2cc(OCC)ncc2)=O)CCN(C(c2sc(C)cc2Cl)=O)CC1C 7902,C(=O)(C(C)CC(F)F)NCC(CC=C)NC(c1ccnc(OCC)c1)=O 7903,Cn1c(C(N2CC(O)(C(F)C(=O)NC3CC(=O)N(O)C3)C2)=O)ccc1C#N 7904,CC1CCCC1(O)CNC(=O)C(c1ccnn1C)NC(c1cnc(C2CC2)o1)=O 7905,c1(C(=O)NC2CCCN(C(C3CN(CC)C(=O)C3)=O)C2)ccc2c(c1)CCCN2 7906,C1(OC)CCC12CC(C(=O)NCCn1cc(CSC34CCN(CC3)C4)nn1)C2 7907,C(c1ccc(F)cc1)=C(C)C(=O)N1CCC1n1cccn1.C12CCN1C(=O)C=CC2 7908,C(=O)(C(C)S(N)(=O)=O)N1C(C(N2CC(CO)C2)=O)(COC)C=CC1 7909,N(C(=NCCC(=C)C)NC1CCN(c2ccc(-n3cncn3)cc2)CC1)CC=C 7910,N1(C(CC(C(C)C)c2ccon2)=O)CC2CCC1C(CNC(C1(CO)CC1)=O)C2 7911,c1(C(N2CC(C)C(CNC(=O)Cc3ccno3)C2)=O)ccc2c(O)ncnc2c1 7912,C(=O)(C1=CC2(CCOC2)C1)NCCN(C(=O)CCc1cnc[nH]1)C 7913,c1(C(=O)NC2CCC3CC2CO3)nc(CNC(C(CC)NC(N)=O)=O)cc(O)n1 7914,c1(CC)cnc(C(=O)NC2CCC(C(=O)N(C(C)CC(C)C)C)C2)nc1 7915,Cc1cc(=NC(=O)C(=O)NCC2(NC(=O)C(O)C3CCCC3)CCC2)[nH]o1 7916,c1(C(=O)NCCC2(OC)CN(C(C3(SC)CCOCC3)=O)C2)cncc(C)c1C 7917,C1(NC(C2(C)CC=CC2)=O)CC2CCCC(C1)N2C(c1cnc(Cl)s1)=O 7918,O=S(=O)(c1c[nH]c2cc(Cl)c(Cl)cc12)N1CCC(c2cccc(F)c2)C1 7919,N1(C2CCN(C(C3CN(C)C3)=O)CC2)Cc2cccnc2N2CCCC2C1 7920,C1(CNC(c2c(CC)nns2)=O)CN(C(c2c(Cl)cnn2CC)=O)CCO1 7921,c1(N2CCN(CCN(C)C(C3CC(=O)NC3)=O)CC2)ccccc1[N+](=O)[O-] 7922,N1(C(c2cnc(CCC)s2)=O)CCCC(C)(NC(=O)CC(C)(C)OC)C1 7923,c1(C(=O)NCCN(C(CC(C)SC)=O)CC(C)O)cc(F)c(F)c(N)c1Cl 7924,c1(CCC(=O)NCC(C)(C2CC2)NC(C(CO)N(C)C)=O)nc2ccccc2o1 7925,N1(C(C)C)CC(NC(=O)C(C(C)(C)C)NC(=O)C=Cc2nnn(C)n2)CCC1=O 7926,C1(CC)CCC(C(=O)NC2CC23CC(NC(=O)COCc2ccncc2)C3)CC1 7927,C(=O)(C(CCNC(c1cccn1C1CC1)=O)OC)NC1(CC#C)CC1 7928,N1(C(C2(OC)CCN(C(=O)C=CC(C)C)C2)=O)CC(=O)NC(C)C1 7929,N1(C(COCC(=C)C)=O)CCC2C(NC(=O)COC(F)(F)F)C2C1 7930,N1(C(C2(CC)CCCCC2)=O)CC(CN(C)C(c2ccoc2)=O)C2(CC2)C1 7931,C(=O)(C(CC(C)C)NC(=O)C(C#N)C(C)C)N(c1ccc(C)cc1)CC 7932,c1(C(C)OC)nc(C(=O)N(CCNC(=O)CN(C2CCSC2)C)C2CC2)cs1 7933,C1(O)(C(N2CCCC(CC(=O)NCC(CC)n3cccn3)C2)=O)CCCCCC1 7934,C1(NC(C2ON=C(C)C2)=O)CCCC2CN(C(c3csc(C(F)(F)F)c3)=O)CC12 7935,CC1(C(=O)NCC2CN(C(c3csc(C4CCCCC4)c3)=O)C2)CC1(F)Cl 7936,c1(CC)ccc(F)cc1C(=O)NCCCCCCNC(c1cc(F)ccc1O)=O 7937,N1(C(C(C)SCC)=O)CCN(C(=O)CCOC(C)=O)CC1CC(F)F 7938,C12(C(N3CC(CNC(COCCOC)=O)C(C)C3)=O)CCC(C1)C(C)(C)O2 7939,c1(C(N2CC(CCNC(C(C)OC)=O)C2)=O)ccc2nc(O)[nH]c2n1 7940,N1(C(=O)Cn2cc(C(F)F)cn2)CC=CC(NC(C2(c3ccsc3)CC2)=O)C1 7941,C(CC(C(C)(C)C)NC(C1CCCN1C1CCCCC1)=O)N(C(C)=O)C 7942,N1(C(CCOCC(C)C)=O)CC2(CCCC2)C1C(=O)NC(C1(O)CCC1)C 7943,N1(C(CNC(C(C)(C)C)=O)=O)CCC(N=[N+]=[N-])(C(=O)NCC2(O)CCCOC2)C1 7944,C1(NC(C(C)n2cncn2)=O)COCC1CNC(c1csc(C(F)F)n1)=O 7945,C1(N(C(C(C)SCCCC)=O)C)C2CN(C(c3cc[nH]c(=N)n3)=O)CC12 7946,c1(C(=O)NCC2CN(C(CCC3C(C)=NOC3=O)=O)C2)nc(O)nc(O)c1N 7947,Cc1cc(C(N2CCC(OC(C)C(N)=O)CC2)=O)c(Br)cc1F 7948,CCC(C)C(O)CC(=O)NC(CNC(=O)CCCCN(C)C)CC(F)(F)F 7949,C1(OC)CCC(NC(=O)CCN(C)C(c2ccc(C)o2)=O)C1 7950,c1(OC)ccc2cc(C(N3CCC(NC(=O)Cc4cnc(C)o4)C3C)=O)[nH]c2c1 7951,C=CC(O)C(=O)N1CCC(C2CCCN2C(=O)Cn2ccnc2C)C1 7952,N1(CC)CC(C(=O)NCC2CCCC2NC(=O)CC2CCCOCC2)CCC1=O 7953,N1(C(C(C(C)C)F)=O)CCC12CN(C(C1(c3ccc(O)cc3)CC1)=O)C2 7954,C1(C)(CNC(c2cnc(NC(C)=O)o2)=O)CCCN1C(c1cnn(C)c1Cl)=O 7955,Nc1ccc(C(=O)NCC2CCN2C(=O)CC2CCCS(=O)(=O)C2)nc1N 7956,C(=O)(CC(CCC)CCC)N1CC(CC=C)(NC(c2cccs2)=O)C1 7957,C(=O)(C1=CC(C)(C)C1)N(C)CC1CCN(C(c2cnc(C)nc2)=O)C1 7958,C(=O)(C(C)(C)C(=O)NCC1CCC(NC(c2cn(C)nc2C)=O)C1)OC 7959,CC1(C)CCCN(C(C2CC(N=[N+]=[N-])C2)=O)C1C(=O)NCC1CCOC1(C)C 7960,c1(CNC(c2cnc(C)s2)=O)ccc(C(=O)NCC2(F)CCOCC2)nc1 7961,C1(O)(Cn2cc(-c3n(C)ncc3)nn2)CCN(C(c2ccc(C(=O)O)[nH]2)=O)C1 7962,C(C1=CCN(C(c2cnc(-c3ccsc3)s2)=O)CC1)NC(CC1(C=C)CCC1)=O 7963,C1(C(N(C)Cc2c(C)cco2)=O)C2CC3C(C2NC(C2CCC(F)C2)=O)C13 7964,C(=O)(C1=CC2CCCC12)N1CC(CCNC(=O)CCc2ccco2)C1 7965,CC(CC(N)=O)C(=O)NCC(C)N(C)C(C1(C(F)(F)F)CC=CCO1)=O 7966,c1(C(N2CC(NC(c3cn(C)[nH]c3=N)=O)CC2(C)C)=O)ccn2nncc2c1 7967,N1(C(C2C(OCC)CC2)=O)CC2OCC(NC(=O)C(F)(F)C(C)(C)O)C2C1 7968,c1(C(N2C3CCC2CC(C(N2CCC(CO)C2)=O)C3)=O)c(F)cc(Cl)cc1Cl 7969,N(C(=NCC1CCC1)NC(c1ncc(C)s1)C)C(C=C)C 7970,C=C(Br)CCC(=O)NCC(CC)N(C(=O)COC(F)F)C 7971,C(N=c1ccnc(CO)[nH]1)C12OCC(CNC(C3CCC(C)CC3)=O)(C1)C2 7972,c1(C(=O)NCC(=O)NC(C)(C)C)ccc2c(c1)C(C)(C)CCN2 7973,c1(CC(=O)NC(CCNCC=C)C(=O)OC)c(C)nn(C)c1C 7974,c1(-c2c(C(N(CCC(C)NC(C3CC3(C)C)=O)C)=O)c[nH]n2)ccccc1Br 7975,C(=O)(C(CC)CC(C)C)NCC(=CC(=O)NC(CC)CCCO)C 7976,c1(C(N(CC(C)(C)NC(C2C(CCC)C2)=O)C)=O)cnsc1C 7977,N#Cc1ccc(Cl)nc1NC(C1C2CN(C(C3CC3(F)F)=O)CC12)=O 7978,C=Cc1ccccc1-c1ccc(CNC(c2sc(C)nc2C)=O)cn1 7979,S(=O)(=O)(c1cccnc1NCCC1CC(C)OC(C)C1)NCS(CCC)(=O)=O 7980,c1(N(CCCNC(C2CNC(=O)N2C)=O)CC)ncnc2c1ncn2C 7981,c1(C(=O)NC2CC3(CCN(C(CNC=O)=O)C3)C2)nc2ncc(Br)cc2[nH]1 7982,C1(CC)CCC(C(=O)NCCOCCN(C(=O)C(C)C#N)C)O1 7983,N1(C(=O)CCC2CC2)CC2CCN(C(C3(C(F)F)CC3)=O)CCC2C1 7984,N1(C(C)=O)CCCC1CC(=O)NC(C1CCCN1C(=O)CC1(C(F)F)CC1)C 7985,Cc1ccc(Cl)cc1NC(c1ccc(N2CCOC(=O)C2)cc1)=O 7986,N1(C(C2CC(C)(C)C2)=O)CCC2CN(C(c3cc(C(C)(F)F)n[nH]3)=O)C2C1 7987,N1(CC(=O)N(C(C)C)CCN(C)C(c2ccc(Cl)s2)=O)CCc2ccccc21 7988,C(=O)(C(CO)NC(c1cn(C)cn1)=O)NCC(C)NC(=O)OC 7989,c1(C(N2CCC(C(N3CC4CC4(CO)C3)=O)C(O)C2)=O)ccc2cncn2c1 7990,c1(C(N2CCN(Cc3cc(OCC)cc(F)c3)C3C2C3)=O)ccc2cnoc2c1 7991,C1(C(=O)Nc2ccsc2CO)CC2(CC2)CN1S(=O)(=O)c1cccs1 7992,C1(C(N2CCCC(CCC)(NC(C=CCCC)=O)C2)=O)CCC2C(C1)C2(F)F 7993,C(=O)(C(C)(F)C(C)(C)F)NC(C)CC1CN(C(C2CCCS(=O)(=O)C2)=O)C1 7994,c1(C(N2C(CCNC(C3CCCCS3)=O)CSCC2)=O)ccc2c(c1)OCO2 7995,Cc1nc(C(=O)NCC(C)(C)NC(=O)CC2C=NN(C)C2=O)sc1C 7996,C1(CNC(Cn2c(C)c(Cl)cn2)=O)CN(C(=O)C2=COCC2)CC(C)(C)C1 7997,N1(C(Cn2ncc(CC)c2)=O)CC(C2CC2)(C(N2CC(C3CC3)OC(C)C2)=O)C1 7998,C1(CC(C)NC(=O)Cc2cnccc2Cl)CCN(C(c2cc(Br)n[nH]2)=O)CC1 7999,c1(OC(C)C(=O)NC(CNC(=O)Cc2csc(Br)c2)C2CC2)cccnc1 8000,N1(c2cn(CC3N(C(=O)NC4C5OC(=O)CC54)CCC3)nn2)CCC(F)(F)CC1 8001,Cc1cc(C(=O)NCC(C)CNC(c2cnc(-c3ccoc3)s2)=O)cc(N)c1O 8002,C1(C(=O)NCCN(C(=O)CSC(F)(F)F)CC)CC2CC(OC)C2C1 8003,Nc1cc(C(=O)NC23CC(CNC(C4CC=CCC4)=O)(C2)C3)ncc1Cl 8004,N1(C(C(C)=CC)=O)CCCC(C2CCN(CC(=O)N(c3nccs3)CCC)C2)C1 8005,c1(C(N2C(CN(C(c3ccnn3C)=O)CC)CCC2)=O)ccnc2ccnn12 8006,N1(C(c2nc(N)c(Br)cc2)=O)CC2(CCN(C(c3ccnn3C3CC3)=O)C2)C1 8007,c1(CNC(c2n(CCCC)nnn2)c2conc2C)nc(C)c(C)cn1 8008,CCC(C)CCC(=O)Nc1ccc(NC(=O)CC2(C)CCOCC2)cc1C 8009,N1(C(C)(C)C)CCC(CC(=O)NC2CC(n3cc(C4CCOC4)nn3)C2)C1 8010,C(=O)(C(CNC(C1(C(C)C)CC1)=O)CC(C)C)NC(c1c(C)nn(C)c1)C 8011,Cc1ccsc1CN(C(c1ccc(F)s1)C(=O)NCCCF)C 8012,C1(NC(c2c(CCCC)ocn2)=O)(COC)CCN(C(c2ccc(C#N)o2)=O)C1 8013,n1(CC)cc(CN(C(=O)CSCCNC(=O)Cc2cc[nH]c2)C)cn1 8014,c1(C(N2C(CCCC)CN(C(c3nccn3C)=O)CC2)=O)cnc2sccc2c1 8015,C1(C)(C(=O)NCC(CNC(c2cnc(Cl)s2)=O)OC)CCCCCC1 8016,C#CCCCCCCCC(=O)N1CC(C)CCC12CC2 8017,CCCCC(CN)NC(=O)C(N1CCC(c2ncc[nH]2)CC1)=O 8018,CC(C)S(=O)(=O)C(C)C(=O)N1CC(C)(C)OCC1CNC(C1(CC2CC2)CC1)=O 8019,c1(NC(C)C)ncccc1C(=O)NCC1CCN(C(=O)C(C(C)O)N(C)C)C1 8020,N1(C(C2C(CC)C2)=O)CCC(C)C(NC(c2cc(-c3ccco3)on2)=O)C1 8021,C(C)(C(=O)N1CC(O)CO1)N(CCC)C(C1CN(C)CCN1C)=O 8022,C1(OC)(CNC(=O)C(C2CC=CCC2)NC(=O)Cc2cc(C)no2)CCCCC1 8023,Cn1cnc2c3c(ccc12)N(Cc1ccccc1F)C(C)C3 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8095,C(C)(C)(C(c1nnnn1C1CCOCC1)NC12CC(C1)C2)OCC 8096,C1(C(=O)NC2CC(NC(c3c(CC)sc(=N)[nH]3)=O)C2)C2CCCCCCC12 8097,C(c1nnn(C)n1)=CC(=O)N(CC(=O)N(CCCN(C)C)CCO)CC.C1CO1 8098,C(CN=c1ncc(F)c[nH]1)C1(O)CCN(C(c2cnc(COC)nc2O)=O)CC1 8099,C1(CC(=O)NC)(CC(=O)NCC2C=CC(NC(C3CC(SC)C3)=O)C2)CCCC1 8100,c1(C(N(C2CCN(C(=O)C(CO)N(C)C)C2)CC)=O)cnn(-c2cccnc2)c1 8101,C1(CC)CN(C(=O)NC2CC3(C2)CC3NC)CCC1c1ccccc1 8102,c1(C(N(C)CCC2CCCCN2C(=O)CC2CC2)=O)nc2ccccc2[nH]1 8103,c1(C(N(CC(CC)NC(=O)CCC2CCCC2)CC)=O)nc(OC)ccc1C 8104,Cc1cc2[nH]c(C(N3CCCCC3C3CCN(c4nnn(C)n4)C3)=O)cc2s1 8105,c1(CC)nn(C)cc1C(=O)NCC1CCCC1NC(=O)COc1ccsn1 8106,C1(CC)CN(C(=O)CN2CCCC2C)CCN1C(=O)Cc1ccc(C)cn1 8107,Cc1ncccc1C=CC(=O)N(C)CCOCCCN(C)C(C1CCOCC1)=O 8108,N1(C(C(C(C)OC)N(C)C)=O)CCC(CNC(=O)CC2OCCCO2)CC1C 8109,C1(NC(C(C)NC(N)=O)=O)C(C)(C)C(NC(C2SCCCS2)=O)C1(C)C 8110,C12(C(=O)NCC3(CNC(CCOCC#C)=O)CCCC3)CCCCN1CCC2 8111,N1(C(c2[nH]cc(C#N)c2)=O)CCC(CNC(c2cccnc2C(F)F)=O)C12CC2 8112,CC1(NC(=O)CC(F)(F)F)CCC(NC(c2cnc(-c3ccccc3)[nH]2)=O)CC1 8113,c1(C(N(C(CCNC(CC(CC)C)=O)C)C)=O)ccc(NC(C)=O)cc1OC 8114,S(=O)(=O)(c1cc(F)ccc1F)N1CCn2c(C)nnc2C1 8115,N1(C(C(CC=C)(F)F)=O)CCN(C(=O)CNc2ccccc2C(N)=O)CC(O)C1 8116,N1(C(CNc2onc(C)c2NC(=O)CC2COCCO2)=O)CCCOC(C(C)C)C1 8117,C(=O)(CCCC(=O)CNC(c1cc(OC)ccn1)=O)NC 8118,c1(CC)cccc(OC(C)C(=O)NC2CC(C)(CNC(c3ncsc3C)=O)C2)c1 8119,c1(C(=O)NC2CCC(NC(C(CSC)O)=O)CC2)ccc(=O)n(CC(F)(F)F)n1 8120,N1(C(c2c(SC)cccc2)=O)CC(NC(=O)CCn2cccc2)CC(O)C1 8121,O=C(N1CC(O)CCO1)NCc1ncc(Br)cc1Cl 8122,c1(OC)ccc(CC(=O)NCC(C)CNC(=O)C(O)C2CCC2)c(Cl)c1 8123,N1(C(c2ccn(CCC)n2)=O)CC(C2(NC(=O)CC3CCCSC3)CC2)C1 8124,C(=O)(N(C)NC(=O)c1ccccc1-n1cc(CNC2(C(=O)O)CCC2)nn1)OC 8125,CC1CN(C(=O)C(C2CCN(C(c3[nH]ccc3C3CC3)=O)CC2)C)C(C)C1C 8126,C1(C(N(CC(CC)(C)OC)C)=O)CC2CC1CC2NC(=O)COC1(C)CCCC1 8127,C(C)(N=c1[nH]c(Cl)ncc1F)C1OCCN(C(C(CCC)CCC)=O)C1 8128,C=Cc1cc(C(=O)NCC2(NC(c3c(CSC)noc3C)=O)CCC2)cc(F)c1 8129,C=CCC(C1CC1)NC(C1CCN1C(=O)CSC)=O 8130,C1(NC(CC(C=C)C)=O)CN(C(c2cccc3ccccc23)=O)CC2(CCC2)C1 8131,N1(C(CCC2C(C)C2)=O)CCOCC1CCNC(=O)CCSC(F)(F)F 8132,N1(C(c2[nH]c(C)c(C)c2C)=O)CC(Nc2ncc3ncnc-3[nH]2)CC(C)(C)C1 8133,c1(CCC)c(C(=O)NCCN(CCOC)C(C2CCOC2C2CC2)=O)cnn1C 8134,C1(C(=O)NC2CC3CC(N(C(=O)C(=O)NC4CC4)C)CC32)CCC2CC1CO2 8135,N1(C(C2(O)CCN(C(C3CCCNCC3)=O)CC2)=O)CCC12CCCCC2 8136,C=CCC(C(=O)NC1(CCOC)CCN(C(=O)CCCCCC)C1)C(C)C 8137,CP1(=O)CCN(CC(=O)Nc2cccc(CNC(=O)Cn3ncnn3)c2)CC1 8138,C#CC1(NC(C2(CNC(=O)C(C)Cn3cccn3)CC3(CC3)C2)=O)CCCOC1 8139,C1(C(=O)NC2C(C)N(C(=O)COC3CC=CC3)CC2)CC2(CC2)CN1C 8140,C12(C(=O)NCCN(C(C(C)OCC)=O)CC3CC3)COC(CC3CC3)(C1)C2 8141,c1(N2CCC(COC)CC2)nc2ccccc2nc1N1CCOC(C)CC1 8142,N1(C(c2cc(C)c(Cl)s2)=O)CC2CCCC2(NC(c2cnc3occc3c2)=O)C1 8143,C#Cc1ccc(C(=O)NCC2CC(CNC(c3ccc(C)cn3)=O)CO2)cn1 8144,c1(C(=O)NCCN(C(C(C)OC)=O)C)ccnn1C1CCC1 8145,C1(C(=O)NCCCOC)CN(Cc2c(F)cc(F)cc2Br)CCC1(F)F 8146,C(CCC(C)(F)F)N(C(CC1(C)CC1)C(=O)NCCc1cccc(F)c1)C 8147,CCCC(C)CCNC(=O)CCNC(=O)C(C)(C)C1CCOC1 8148,c1(C(CNC(C23CC2CCN3C(C)=O)=O)OCC)cccc2ccccc12 8149,C=C(CCC(=O)OC)C(=O)NC1CNCCNC1 8150,Cc1cc(-n2cc(CSCCNC(=O)CC3CCC(C)(C)CC3)nn2)ccc1N 8151,c1(OC)ccc(C(=O)NCC(C2CCCN2C(c2n[nH]c(C)c2F)=O)(C)C)cn1 8152,C12(CNC(c3cc(C)on3)=O)CCC(CC1)N(C(c1cc3ccccn3c1)=O)C2 8153,c1(C(=O)NCCN(C)C(C2CC(S(C)(=O)=O)C2)=O)ccc(N)c(Cl)n1 8154,Cc1ccnc(NC(=O)C(C(C)C)NCCC2CC3CC3O2)n1 8155,c1(OCCCCCOc2ccc(F)cc2)cnc2cccnn12 8156,c1(CC(=O)OCc2ccc(OCC=C)cc2)c[nH]c2cccc(C)c12 8157,N1(C(CC2CNC(=O)O2)=O)CCCN(C(=O)CNC(=O)CC(F)(F)F)CC1 8158,C1(NC(CC2(C)CC(F)(F)C2)=O)Cc2ccccc2N(C(c2csnc2Cl)=O)C1 8159,CC1CC(C(=O)N(CCCCCC(=O)N2CCCCC(C(=O)N(C)C)C2)C)=NO1 8160,C1(C(=O)NC(C(=O)NC(C2(O)CCCCC2)C)CC2CC2)CC2(CCC2)C1 8161,C(C)(C)(CC(=O)NC(c1ccc(F)cc1)CNC(=O)CSC1CC1)SC 8162,n1(CC)ccc(CNC(=O)C(C)N(C(=O)CCC2(C)CC2)C2CC2)n1 8163,N(C1CCC(N=c2cc(C)c(C#N)c[nH]2)c2ccccc21)C(c1c(C)ccs1)=O 8164,c1(OC)ccccc1C(CNC(=O)CCC(C)SC)NC(C12CC(CO1)C2)=O 8165,N1(CC(=O)NCC2C(NC(CCCc3nnc(C)n3C)=O)C2)CCc2sccc2C1 8166,c1(C(N2CC(CC(C)NC(CC(C=C)(C)C)=O)C2)=O)ccc2c(c1)ncn2C 8167,Cn1c(O)ncc(C(=O)NCC2(NC(C3CNC(=O)N3)=O)CCOC2)c1=O 8168,CCCC(C)N(CCC(=O)NCC(C1CC1)N(C(=O)C(O)C1CCCC1)C)C 8169,C12(NC(C3CC(C)(F)C3)=O)CCCCCC1N(C(c1cc(O)ccc1Cl)=O)CC2 8170,c1(C(N(CC(C)NC(=O)Cc2cncnc2O)C)=O)ccnc(Cl)c1Cl 8171,N1(C(CC2(C=C)CCCCC2)=O)CC2CCN(C(C3SCCS3)=O)C2C1 8172,c1(-c2cn(CC(=O)NCC3(O)CC3)nn2)ccc(C(F)(F)F)cc1 8173,C(=O)(C(CC)C(=O)N1CCCC(NC(=O)CCCc2ccc(C)cc2)C1)OCC 8174,N1(C(c2cn(C)nc2)=O)CCN(CC(=O)NCCN2CC=CCC2)CC1 8175,c1(C(=O)NC23CN(C(C(CCCC)C)=O)C(CC2)CC3)c[nH]c2c(F)cccc12 8176,C1(C(=O)NCC2CC(OC)C2)C2CC3C(C2NC(c2cc(C)nnc2C)=O)C13 8177,N1(C(C(C(C)C)NC=O)=O)CC2(C1)CN(C(C1CC1C(C)O)=O)CC2CO 8178,Cc1c[nH]c2ncc(C(=O)NCC3(CNC(=O)CN4CC5CCC4C5)CC3)cc12 8179,C=CC(C)(C)C(=O)N(CC(O)CN(C)C(C1(CC)CCOC1)=O)C 8180,C12(NC(=O)CCF)CCCC1CN(C(c1ccc(-c3ccsc3)nc1)=O)C2 8181,c12cccnc1NC1CCC(C1)NC2=O.C1(C(=O)NC(C)C)(CC2CC2)CC1 8182,c1(C(=O)NC2C(CNC(=O)CCF)COC2)ncccc1C1CC1 8183,c1(OC)ncc(C(=O)NC2(CN(C)C(c3ccn(C)c3)=O)CC2)cc1C 8184,C1(C)(C(=O)NCC2CC(NC(c3n(CC)ccc3)=O)C2)CCC(=O)N(C)C1 8185,CC1CN(C(=O)COC2CCC2)CCCN1C(C1C2COCC12)=O 8186,C1(N(C(Cn2nnc(=N)[nH]2)=O)CCO)CCN(C(=O)CC2CC(OC)C2)CC1 8187,c1(CC)nc(OC(C2CN(C(=O)COCC3CCCC3)C2)C)cc(C)n1 8188,C1(NC(c2coc(Cl)n2)=O)CCC2(CC1)CCN(C(c1ccc(I)c(O)c1)=O)C2 8189,C(C)(N=c1[nH]c(=N)[nH]c(=NCC(C)C#N)[nH]1)c1c2nc(C)oc2ccc1 8190,c1(C(=O)NC2C(NC(C(C)Sc3nc[nH]n3)=O)CCC2)cccc(C(F)(F)F)c1 8191,C1(C(N2CCC(O)(CNC(C=C(C)Cl)=O)CC2)=O)CC1C1CC(F)(F)C1 8192,N1(C(c2cnc(CCC)s2)=O)CC(NC(=O)C(C)(CC)CO)C(C2CC2)C1 8193,CC1(C)COc2ccc(C(=O)NC3CN(C(c4cc(Cl)no4)=O)CC3O)cc21 8194,Cc1nnc2n1C(C(=O)N1CC(C)(NC(C3CCc4ncncc4C3)=O)C1)CC2 8195,C1(C(=O)NC(C(=O)OCC)CC)CN(C(C2(Cl)CCC2)=O)CC12CC2 8196,C1(NC(C=CCCC)=O)CCC2(CCN(C(C3(C)CCCC3O)=O)C2)C1 8197,C1(O)(CNC(c2n(C(CC)C)ncc2)=O)CCN(C(C2CCCOCC2)=O)CC1 8198,Cc1cnn(C)c1C(=O)NCC=CCNC(C1CCCN(c2ncccn2)C1)=O 8199,C1(NC(=O)CBr)CCC(CNC(C2(n3cccn3)CC2)=O)C1 8200,C(C(C(=O)N(C)CC1CCN(C)C1)C(C)(C)C)NC(C(C)(C)SC)=O 8201,c1(OC)nc(C)cc(C)c1-c1noc(C2CCCN(C(C)=O)CC2)n1 8202,C(C)(C)(CCCC(=O)Nc1cnn(C)c1C)NC(CCn1ccc(C)n1)=O 8203,C12(C(=O)NC3CCN(C(CC(C=C)C)=O)C3C)CCC(CC1)C(C)O2 8204,C1(NC(=O)CN2CCCC2=O)CC2CC1N(C(c1nccc(F)c1Cl)=O)C2 8205,c1(SCC(=O)NCC(C)NC(c2ccc(OCCF)cc2)=O)ccc(O)cc1 8206,N1(C(C=COCC)=O)CCC2(CC1)C(NC(=O)CC1CC1(C)C)CS(=O)(=O)N2C 8207,N1(C(C2N(C(c3nn(C)c(F)c3)=O)CCCC2(C)C)=O)CCC(C2CCCC2)C1 8208,c1(CC)c(C(C(=O)NCc2nnn(C)n2)N(CC(C)CO)C)cccc1C 8209,N1(c2ccnc(NC(c3ccncc3Cl)C)n2)CC2CC1CS2=O 8210,N12CCCN(CC1)COC(Cc1cnc[nH]1)C2=O.C(=O)(CC(=O)OC(C)=O)NCC 8211,Cc1cc(C(N2CCCC2CCCNC(=O)Cc2ccsc2C)=O)[nH]c1C 8212,CC(C)(C#CC(=O)N1CC(O)C(C)(C)C1)CNC(C1CCC(=O)CC1)=O 8213,Cc1cc(C(=O)NC(C2CCN(C(c3ccccc3Br)=O)C2)C)ccn1 8214,c1(NC(CNC(C(N2CCC(C)C2)=O)=O)=O)c[nH]c2cccc(Cl)c12 8215,N1(C(CCC#N)=O)CCN(C2CCCC2NC(=O)CC(O)CC2CC2)CC1 8216,c12cc(n[nH]1)NC(=O)OC2.N1(CC(C)=CC(=O)OC(C)(C)C)CCOCC1 8217,C1(CCCC)(C(N2CCC(C(=O)OC)C2)=O)CN(C(C2CCC2C(=O)OC)=O)C1 8218,c1(C(=O)NCC2CCC(CC(=O)OC)CC2)cc2cccc(Br)n2c1 8219,C1(C(=O)NC(C)CC(=O)N(C)CCOCCCO)CC2CC(=O)C1O2 8220,C1(C(N(c2nccs2)CC)=O)CCN(Cc2ccc(F)s2)C1 8221,c1(CNC(=O)NC)ccc(Cl)c2cc(CCOCCOC(=O)OC(C)(C)C)[nH]c12 8222,C1(CC(=O)NCC2(NC(C3CCC4(CCC4)O3)=O)CCCC2)CCC2(CCC2)O1 8223,C(=O)(CCC(=O)NCCC1COCCN1C(=O)Cn1cc(C2CCC2)nn1)NC 8224,C(C(C)(C)N=c1[nH]nc(C#N)s1)N(C)C(c1cc2c(=O)[nH]ccn2n1)=O 8225,C12(CN)CCCC1CN(C(C1CC3(CO1)CN(Cn1ccncc1=N)C3)=O)C2 8226,N1(C(c2ccc(NCC)cc2)=O)CCC2(CNC(=O)C(O)C(C)C)CCCCC12 8227,c1(C(=O)OC)cc(C)cnc1NC1CC(C)N(C(c2cnn(C3CCC3)c2)=O)C1 8228,C(CC(C)C)(C(=O)N1CCC(C(C)CO)CC1)N(C(CSCCC(C)C)=O)C 8229,N1(C(Cc2cnn(C)n2)=O)CC2(CCC(CNC(c3ccc(C4CC4)s3)=O)O2)C1 8230,C1(C(=O)NCCCC(=O)NCCCOCC=C)CC(=O)OC1(C)C 8231,C(=O)(C1=C(F)CN(C(C2CC3(CC3)CO2)=O)CC1)N(C)Cc1cncn1C 8232,c1(SC)cc(C(=O)NC2COCCN(c3ccnc(C)n3)C2)ccc1[N+](=O)[O-] 8233,c1(C(N2CC(c3ccccc3)C2(C)C)C(=O)NC(C)C)cc(C2CC2)ccc1F 8234,C1(NC(C2CCN(CC(C)C)C2)=O)CN(C(=O)CCCC2CC2)CC1O 8235,C1(CNC(c2c(C)cc(C)s2)=O)CCC12CCN(C(C1CCCOC1)=O)CC2 8236,N1(C(c2cc(I)cn2C)C(=O)NCCCC)CCOc2cccc(F)c2C1 8237,N1(C(COCC)=O)CC=CC1(C(=O)NC1CCC2(CC2)C1)COC.N1CC(O)C1 8238,c1(C(C)NC(=O)NCc2sc(C)cc2Br)cnc(Oc2ccccc2)cn1 8239,Cc1ccc(-n2cc(CCCNC(C3(C(F)(F)F)CC3)=O)nn2)cc1Cl 8240,c1(C(=O)NCCN(CCOC)C(C2CN(c3nncs3)C2)=O)cc(CO)n(C)n1 8241,Cc1c[nH]nc1C(=O)NC(C)CC(C)NC(=O)C(c1cncnc1)C 8242,C(=O)(C1=CCCCO1)NCCN(C(C1(O)CCN(C(=O)OC(C)(C)C)C1)=O)CO 8243,c1(CC(=O)Nc2cc(Cl)c(Br)cn2)c(F)ccc(Br)c1F 8244,C1(CCC(=O)NC2CCCC2CNC(C2CC(=O)N2)=O)CCCCO1 8245,C(=O)(CC(C)CNC(C1C=CCCN1C(=O)CSC(C)(C)C)=O)OC 8246,c1(C(N2CC(OCC)(CNC(=O)C(C(C)(C)C)SC)C2)=O)cnc2nccn2c1 8247,Cc1cn(C)nc1C(N1CCC(CNC(=O)CC2CCC(C(F)(F)F)O2)CC1)=O 8248,C(=O)(C(C)(C)c1cccnc1)NCCN(C(C)C)C(c1nocc1Br)=O 8249,C1(NC(c2c(OC)csc2)=O)C2CC(O)C1N(C(=O)C=CC1C(C)C1(Cl)Cl)C2 8250,c1(C(=O)NCCCCCCNC(C2N(CC)CCC2)=O)[nH]c(=N)ccc1C 8251,CN1CCN(C)C(CN(C=O)Cc2ccc(-c3cccc(Cl)c3)o2)C1 8252,C1(C(N2CC(NC(c3cncnc3)=O)C(O)CC2)=O)CC2CC1CC2(F)F 8253,N1(C(c2c(CC)con2)=O)CC=CC(C(=O)NCC#CC2CC2)C1 8254,c1(CC(N2CCC(C(CNC(C(CC#C)C)=O)(C)C)CC2)=O)ccc(Cl)c(F)c1 8255,c1(-n2cc(C3N(C(CSC(C)(C)C)=O)CCC3)nn2)ncc(Cl)cc1Cl 8256,CC1COCC(C(=O)NC(C)(C(=O)NCC2(N(C)C)CCCC2)C2CCC2)O1 8257,C1(C(=O)NCCN2CC(=O)NCC2)C2CCC(C2)C1NC(C1CC(=C2CCC2)C1)=O 8258,c1(C(C(=O)Nc2c(C(=O)OCC)c[nH]n2)(C)C)ccc(Cl)cc1Cl 8259,C1(=O)C(CC(F)(F)F)Cc2cn(nn2)C2COCC2N1.CC(C)(CO)CCCO 8260,C(=O)(CCCC(C)(C)NC(=O)C(C#N)C(C)C)NCC(CC)(C)CO 8261,c1(CN2CCC(C(N3CCCCC(F)(F)CC3)=O)CC2)cncc2ccccc12 8262,C=CCC(CC=C)C(=O)NC(C)(C)CCNC(c1cn(C)nc1C(F)(F)F)=O 8263,Cc1ccc(C2(NC(=O)CCOCC(=O)NC(C)CC3CCOC3)CC2)nc1 8264,CC1CCC(NC(=O)CCCC2CC2)CN1C(=O)CNC(N1CCCC1)=O 8265,O=S(=O)(c1ccc(NCc2ccc(-n3cccn3)nc2)cc1)C(F)(F)Cl 8266,C1(CNC(C2(CC#C)CCCC2)=O)CC(NC(c2cc(Cl)ccn2)=O)C1(C)C 8267,C(CC(C)(C)C(=O)NCC(c1ccccc1)CNC(C1(F)CC1C)=O)SC 8268,NC(CCC1CCC1)C(=O)NNc1cc(F)ccc1Br 8269,C(CCC(C)(C)NC(=O)CC1CCC(C)C1)NC(CSc1nc(C)[nH]n1)=O 8270,C(CS(=O)(=O)CC(=O)NCCC1(NC(=O)CN2CSCCSC2)CC1)OC 8271,N1(C(C2(C)CC(C)C2)=O)CCN(C)C(CNC(C2(C)CCCS2)=O)C1 8272,C(C(=O)NOC1CC2CCC1C2)(c1ccco1)NC(C1CC1(Cl)Cl)=O 8273,C1(NC(CCC=C)=O)CC2CCCC(C1)N2c1cc(SC)ncn1 8274,C1(NC(CC2CC(SC)C2)=O)C=CCN(C(c2ccc(C)cn2)=O)C1 8275,CCCCC(C(=O)NCC1CCCN(C(c2ncccc2CO)=O)CC1)C(C)C 8276,C(CCCCCCCO)=CC(=O)NC1CN(C(C(CSC)C)=O)CC2C1C2 8277,C1(NC(C2(CC)CCC2)=O)CN(C(c2ccc(C(N)=O)cn2)=O)CC1C 8278,c1(C(N2CCCC(O)(CNC(C(C(C)C)C#N)=O)C2)=O)sc2cccnc2c1Cl 8279,N1(C(C(C)O)=O)CCCC(C2CCCN(CCCOc3cccc(Cl)c3)C2)C1 8280,C1(C(=O)NCC2(C(=O)NCc3n(CC)cnc3)CC3(CC3)C2)CC2(C1)CC(C)C2 8281,C1(C(N2CC(C(C)OC)C2)=O)(CCNC(=O)C(C)C2CC2)CCCC1 8282,c1(C(=O)NC2CC(F)(CNC(CCOCCCOC)=O)C2)cccnc1C(F)F 8283,c1(OC)cc(OC)cc(C(=O)NCCC2CCN(c3nncs3)C2)c1 8284,C1(NC(CN(C(COC)=O)C)=O)CC(F)CN(C(=O)C(F)(F)CO)C1 8285,c1(CCNC(C(N2CCC(C(N)=O)CC2)c2cn(C)nn2)=O)cccc(F)c1 8286,C1(CNC(C2(CCC=C)CC2)=O)CC2CC1CN2C(=O)COC(C)CC 8287,c1(C(=O)NC2CC3(C2)CN(C(=O)COCC2CC2)C3)cc2cccc(F)c2s1 8288,CN1CCC(=CC(=O)NCC2CCN(C(=O)CC3CCC(=O)N3)C2)CC1 8289,C(=O)(C(C)(C)C(F)F)N(CC(C)(C)NC(C1CC12CC2)=O)C 8290,c1(C(N2C(C)CN(C(C3(C)CCC(=O)N3)=O)CC2)=O)ccc2ccccc2n1 8291,N1(C(C2CN(C(c3c(C)nsc3C)=O)CC2C)=O)CCCc2occc2C1 8292,C1(CC(=O)NCC2C(C(=O)NCC(COC)(F)F)CCO2)C(=O)NN=C1C 8293,C12(CNC(COCCCOCC)=O)CC(NC(=O)CC3COCCO3)(C1)C2 8294,C1(C(N2CC(CCNC(c3cc4cn[nH]c4cn3)=O)C2)=O)CC2CCCC(C1)C2 8295,Cc1ccsc1C(=O)NCC1C=CC(NC(=O)C(O)CC2CCOCC2)C1 8296,c1(C(C)C)ccc(-c2nc(C3CCCC(n4cccc4)C3)n(CC3CC3)n2)cn1 8297,C(C(CC(F)(F)F)NC(C1(O)CC1)=O)NC(c1nc(CC(C)C)sc1)=O 8298,N1(CCCC2CCCCC2O)CCC(CCCl)CC1.C12CC1C(=O)NC2=O 8299,N1(C(CN(C2CCC2)C)=O)CC2CCC2(CCNC(=O)C=Cc2nccs2)C1 8300,c1(C(=O)OC)cncc(-n2cc(CONC(c3ccnnc3O)=O)nn2)c1 8301,N(C(=NCCC(C)SC)NC1CC1NC(=O)OC(C)(C)C)C1CC(OC)C1 8302,Cc1ccc(CC(=O)NCC23CC(CO2)N(C(C2CCC(C)C2)=O)C3)cc1C 8303,C1(C#N)(C(=O)NCC(C)NC(C2N(C(C)=O)CCC2)=O)CCCOC1 8304,C1(CC(=O)NC(C)C(C)n2cccn2)C(NC(=O)Cc2cncs2)CC1O 8305,N1(C(c2n(CC#C)cnn2)=O)CCC(C)C1C(=O)NC(C)(C)C#CCC 8306,c1(CC)ccc(C)c(C(N2CCC(CCNC(C3SCC=C3C)=O)CC2)=O)c1 8307,c1(C(=O)NC2C(CNC(c3ccc(O)cc3)=O)C2)cccc(Cl)c1[N+](=O)[O-] 8308,C1(CC(=O)NC)CCCN1C(C1(C(=O)OC(C)(C)C)CCC1)=O 8309,c1(OC)ncc(Cn2nnnc2N2CCOCC2C(C)C)cc1F 8310,N1(C(C(c2cnccn2)C)=O)CCC(C)C1CNC(=O)CCCn1cccn1 8311,Cc1cnc(C(=O)NC2C3CC4C(C3)C24C(=O)NC(C)Cc2nc[nH]n2)c(C)c1 8312,c1(C(N2CCC(CC)C2CNC(=O)CSC)=O)ccc(F)c(Cl)c1 8313,N1(C(c2cc(C3CC3)ccn2)=O)CC2OCCN(C(c3sccc3Cl)=O)C2C1 8314,N1(C(CCOCC(C)C)=O)CCC(O)C1C(=O)N(CCO)CC1CC1 8315,C(CC(CC)(CC)NC(c1ccnc(OC)c1)=O)NC(C(C)OCC=C)=O 8316,N1(C(c2ccc(CNC(C(CCCC)F)=O)o2)=O)CCC2(CCCOC2)C1 8317,c1(C(=O)NCC(CC)NC(c2oc(C3CC3)nc2C)=O)cnc2c(c1)CCOC2 8318,C1(CNC(=O)NC(C(C)c2ccccc2)(C)C)CC(C)(C)CO1 8319,C12(CNC(C(c3ccn(C)n3)C)=O)CC(CCO1)N(C(=O)CN1CCSCC1)C2 8320,C(=O)(C(C(=O)N1CCC(CNC(=O)C(C)=C(C)CC)C12CC2)C(C)C)OCC 8321,c1(C(N(C2CCCC(NC(=O)Cc3nccn3C)C2)C)=O)ccnc(CO)c1 8322,c1(C(=O)NC2C3CN(C(c4n[nH]c(C)c4C)=O)C(C3)C2)csc2c1CCCC2 8323,N1(C(C2(OC)CC(C)C2)=O)CCN(C(=O)CCn2nc(C)cc2C)CC12CCC2 8324,C(=O)(C(C)(O)C1CCCCC1)N(CCCNC(C=CC=CC)=O)C 8325,C1(CNC(CC2(C)CC2(Cl)Cl)=O)C2CN(C(c3ccc(N(C)C)nc3)=O)CC12 8326,N1(C(C2OCCN(C)C2=O)=O)CCC2(CCC2)C(NC(c2ncccn2)=O)C1 8327,c1(OC)c(C(N2CCCC(NC(=O)C(O)P(C)(C)=O)C2)=O)cccc1Cl 8328,C1(C(=O)NC(c2ccc(O)nc2)C)CC(NC(C2(C)CNC(=O)C2)=O)C(O)C1 8329,c1(C(=O)NC2CCN(C(CCCCNC(N)=O)=O)C2)ccc(N)cc1C(F)(F)F 8330,C1(CNC(C(C)OCCC#C)=O)CN(C(=O)Cc2csnc2C)CCC1(F)F 8331,C(=O)(CC(C)(C)C#N)NC(CC(=O)NCCC(C(C)C)NC(N)=O)c1cccs1 8332,N1(C(C(C(C)C)SC)=O)CC2(CCCN(C(=O)C(c3nc(C)cs3)C)C2)C1 8333,N1(C)CCCOC(CCS)C1.CC1(C)C(N)(C(=O)C)CO1 8334,C1(NC(C(C)N(C(=O)CC2CCOC2)CCC)=O)CCc2c[nH]nc2C1 8335,C(=O)(CC(C)(C)CCOC)NC1(CC=C)CCN(C(=O)C(C)(C)C(C)(C)O)C1 8336,N1(C(c2ncsc2C(F)(F)F)=O)CC2(CCN(C(C3(O)CC4CCC3C4)=O)C2)C1 8337,CC(C)C(O)CC(=O)NCC1CN(C(=O)CCNC(N)=O)CC1C(F)(F)F 8338,CC(C)CC(O)C(C)C(=O)N(C)CCOCCNC(=O)CCC(F)(F)F 8339,C(=O)(C#CC(C)(C)CNC(c1c[nH]cc1C1CC1)=O)NCc1n(CCC)ncn1 8340,N1(C(C(C)c2ccsc2)=O)CCCC(CO)(NC(=O)CO)C1 8341,C1(NC(CNC(N)=O)=O)CN(C(=O)COCc2ncc[nH]2)C2(CCOC2)C1 8342,CC(C(=O)NCC1CCC1C(N1CCN(C)CC1C1CC1)=O)C(C)(C)C 8343,C(=O)(CN=c1cc[nH]cc1)NC1(C)CC(C(N2CC[Si](C)(C)C2)=O)C1 8344,c1(CNC(C(=O)NCCc2cccc(OCCO)c2)=O)cc2cccnc2[nH]1 8345,Cc1cc(Br)cc(C(=O)NC2CC(NC(=O)CCS(C)=O)C2)c1F 8346,C1(C(=O)NC(C2CCN(C(=O)C(F)=C3CCC3)CC2)(C)C)CC2(CC2)CO1 8347,Cc1onc(Br)c1C(=O)N(C)CC1CCCN1C(C1(C)CC(F)C1)=O 8348,N1(C(CCNC(=O)C=CCl)=O)CC2CN(C(=O)CCn3cncn3)C2C1 8349,N1(C(c2n(C=C)ncc2)=O)CCCC2(C1)CN(C(C1CN(C)CC(C)O1)=O)C2 8350,c1(C(C)(C)C)ccc(NC(=O)CC2CC(NCc3c(Cl)cccc3Cl)C2)c(Br)c1 8351,C1(C(N2CC(C(CC)C)C2)=O)CCC(NC(=O)C(C)O)CC1 8352,CC1CN(C(c2cc(C(N)=O)cs2)=O)CC(C)CN1C(c1ccc(N)c(N)n1)=O 8353,CCCCCC(C)CC(=O)NC1CCN(C(c2cccc3c2CCC3)=O)C1(C)C 8354,C1(C(N2CC(C(N3CC(COC(C)=O)C3)=O)OCC2)=O)CC2(CCC2O)C1 8355,NC1CCC2(CC1)CN(Cc1cn(CCc3cccnc3Cl)nn1)C2 8356,CCCCC(CC)CC(=O)NCCCC(C)(C)C(=O)NCC(C)(O)COC 8357,c1(OC)cc(OC)cc(CC(=O)NC2(CN(C)C(C3COC(C)C3)=O)CC2)c1 8358,c1(C(=O)NC(C=C)COC)ccncc1-c1cccc(C(=O)NC)c1 8359,c1(C(N2C(CNC(C3CC3c3cnc[nH]3)=O)CCC2)=O)ccc(C(F)(F)F)cn1 8360,CN1CCC2CN(C(C3CN(C(c4ccc(O)cc4O)=O)C3)=O)CC2C1 8361,c1(C(=O)NC2CC(C(=O)NC(CCCC)CO)OCC2)ccc(=NC)[nH]c1 8362,CCC(O)C(C)C(=O)NCCC1(OC)CN(C(C2CC2F)=O)C1 8363,CC1(C)Cc2[nH]nc(C(N3CCC(O)(CNC(=O)C4=NOCC4)C3)=O)c2C1 8364,CCC(C(=O)NCCCCCN(C(=O)C(C)c1cccs1)C(C)C)C(C)C 8365,N1(C(=O)OC(C)(C)C)C(CC#N)COC1(C)C.c12c[nH]nc1CN(C=O)C2 8366,C1(CNC(c2nn(Cc3n(C)ccn3)c(C(F)(F)F)c2)=O)CC(C2CCC2)C1 8367,C1(OC)CC2(C1)CC(C(=O)NCC(c1ccc(C)cc1)NC(=O)C(O)C(C)C)C2 8368,n1(CC)cc(C(=O)N(CCCN(C)C(C2(C)CC3CC3C2)=O)C)c(C(F)(F)F)n1 8369,c1(C(=O)NCC2(NC(CN3CCCC(CC)C3)=O)CC2)c(F)ccc(N)c1F 8370,c1(C(=O)NCCCCCN(C(C(COCC)C)=O)C)cc(OC)n(C)n1 8371,Cc1cc(C(=O)NC2CC(CCNC(C3(O)CCC(C)CC3)=O)C2)nc(C)n1 8372,c1(C(N2C(CNC(C(C)(C)N(C)C)=O)CC3CC32)=O)cc2n(n1)CC1(CC1)C2 8373,N(C(=NCC(=C)C)NC1CCN(c2ccccn2)C1)C(c1csc(C(F)(F)F)n1)C 8374,C(=O)(C1OCCc2c(Br)cccc21)NC1(CNC(c2cocn2)=O)CC1 8375,O=C(C1CCc2ccccc21)N1C2CC1CN(Cc1c(Cl)cncc1Cl)C2 8376,Cc1cc(C(=O)N(CC(C)O)CCNC(=O)CCC2CCCN(C)C2)cc(Cl)c1 8377,c1(CC)occc1C(=O)NC(C(=O)NCCC(O)C1CC1)C1(C)CC1 8378,C1(CNC(COCCCC(C)C)=O)(NC(=O)Cc2csnn2)CCCCCC1 8379,Cc1cc(N(C)C)nc(C)c1.c12cnc(cc1C)n(C1CCNCC13CC3)c2=O 8380,N1(C(Cn2ncc(CC)c2)=O)CCC2(CC2NC(=O)CCCCON(C)C)C1 8381,N1(C(c2c(CC)nc(C)nc2)=O)CC2CC(NC(=O)CC3CCNC3=O)CC2C1 8382,c1(C(N2CC(CNC(C(CC)(C)O)=O)OCCC2)=O)cc(Br)c(F)cc1F 8383,c1(C(=O)NCC(C)NC(=O)C(c2ccc(Br)cc2)O)cc2c[nH]nc2s1 8384,c1(C(N2CC3C(CNC(C(C=C)C)=O)(CC3)C2)=O)cnn2c1OCCC2 8385,CCC(=O)CCC(=O)N1CC=CC1(C)C(=O)NC1CNC(=O)C1(C)C 8386,C=CC1(CC(N2CCC(C)C2CNC(c2cc(C)cc(C)c2)=O)=O)CCCCC1 8387,C1(CC(=O)NCC2(C=C)CCC2)CN(C(C2CCC2(F)F)=O)CC12CC2 8388,C1(C(=O)Nc2ncc(Br)s2)CC12CCN(C(c1ccno1)=O)C2 8389,O=C1CCC(C(=O)NCC2(CO)CCN(C(=O)CCc3cncnc3O)C2)CN1 8390,Cc1ccc(Cl)cc1NC(=O)CC1CC(C)(C)CN1C(=O)C(C)N=[N+]=[N-] 8391,C1(C(N(CCNC(CC(C=C)C)=O)C2CC2)=O)CC1C1CCOCC1 8392,CCCC(C)(CCC)C(=O)NC(C)CN(C(=O)Cc1ncoc1C)C 8393,CC(CS(C)(=O)=O)NC(c1ccc(CNC(=O)CN(C)C(N)=O)nc1)=O 8394,c1(C(N(CCNC(C(CCC)C(C)C)=O)CCC)=O)cnc2ccccn2c1=O 8395,C1(C2CCN(C(C3CC34CC(O)C4)=O)C2)(NC(=O)CCN2CCCC2)CC1 8396,N1(C(C(C(C)C)C)=O)CC2(CCCCN(C(=O)C(C)(C)C(C)(F)F)C2)C1 8397,Cc1cc(O)ccc1C(=O)NCC(C1CC1)N(C(=O)C=Cc1cscn1)C 8398,N1(C(c2cn(CCC)nc2C)=O)CCC(NC(c2cnnc(C)c2)=O)CC1C 8399,CC(C)(C)C(C(=O)N1CC(C(F)(F)F)C(CNC(=O)CC2CSC2)C1)NC(N)=O 8400,c1(OC)ccc(NC(=O)C(C2CN(C(=O)CC3CNC(=O)O3)C2)SC)cc1C 8401,c1(CNC(C(=O)Nc2c(OC)c(F)c(F)cc2)=O)ccc(Br)c2cccnc12 8402,Cc1cc(C(=O)NC(C(=O)N(C)Cc2cscn2)C2(C)CC2)nn1C 8403,N1(C(C(=O)NCCc2cc(OC)c(C(C)(C)C)cc2)=O)CCC2(CNC(=O)C2)C1 8404,C1(NC(c2csc3nnsc23)=O)CCCCCN(C(C2CCCCC2)=O)C1 8405,CCCCCCCCCCCC(=O)N(C(C)CNC(C1CC(CC)(CC)C1)=O)C 8406,c1(COC)cc(C(=O)OCC(=O)NCc2ccccc2)n[nH]1 8407,C1(CC(N2CCCC(CNC(C(CC)(C)C#N)=O)C2)=O)CCC2(CCCC2)CC1 8408,c1(OC)cnc(C(N2CC(F)(C(=O)NCc3ccc(C)cc3OC)C2)=O)c(F)c1 8409,C(=O)(C(C)(C)C(F)F)N(C1CCN(CC(=O)OC)CC1)CC12CCOC1CNC2 8410,C=CCC(CC=C)C(=O)NCC1CCC1NC(C12CCC(CC1)CO2)=O 8411,c1(C(C)(C)C)cncc(C(N2CCC(F)CC2)C(=O)NC2CCOCC2)c1 8412,c1(COCC)ccc(CO)o1.C1(=O)C(CSC)N1.C12CCOC1c1cnn(c1)C2 8413,C1(C(C(C(=O)NC)C#N)=O)C2COC(C)(C)OCC12 8414,c1(C(=O)NCC(C)OCC#C)coc(CNC(=O)CCC2CC2(F)F)n1 8415,C1(=CCNC(C2CC=CCC2)=O)CCN(C(c2cccnc2C(F)(F)F)=O)CC1 8416,C(=O)(C1=C(Cl)CCOC1)NCC1C(C)CN(C(=O)C=Cc2cccn2C)C1 8417,C12(C(N3CCC(CC(C)NC(C(C4CC4)OC)=O)CC3)=O)CCC(CC1)CO2 8418,c1(CNC(N(C2CCC2O)CC)=O)csc(C2CCCO2)n1 8419,C(CCC(C)C)=CC(=O)N(CC(CNC(C(C)OCC=C)=O)O)C 8420,CC(C)CC(C)(O)c1cn(C2(C(=O)NCC3CCCC3(F)F)CC2)nn1 8421,N#CC1(C(=O)NCc2nc(C(N3CCC(C(F)F)CC3)=O)co2)CCCOC1 8422,C1(NC(Cc2c(C)cc(C)s2)=O)CCN(C(=O)CCC(C)(C)C)C(C)C1 8423,C(=O)(C1=CC2C=CC(C1)C2)NCC(CC(C)C)NC(c1ccccc1C(F)F)=O 8424,c1(C(=O)NCC23N(C(CCOCC)=O)CCC2CC3)cnc2c(c1)CCCO2 8425,CCCC(C(O)C(=O)NCCC(C)C(C)CC)NC(C1(c2ccccc2)CC1)=O 8426,Cc1noc(N)c1C(=O)NCC#CC(=O)NC(c1cncc(F)c1)C 8427,c1(C(N2CCCC(CNC(C(C)OCC=C)=O)C2)=O)c(OC(F)F)cccc1Cl 8428,c1(NC(=O)NCCC(N2CCOCC(N3CCCC3)C2)=O)nc2ccccc2s1 8429,c1(C(N2C(C)(C(=O)NC(CCOC)C(C)C)C=CC2)=O)cc(C)cc(O)n1 8430,N1(C(Cn2cc(CNC(c3n(CC)ccc3)=O)nn2)=O)CC(C(N)=O)C2(CC2)C1 8431,c1(OC)ccccc1C(C)C(=O)N(CC(C)CNC(c1nocc1C)=O)C 8432,N1(C(C(=O)NC(N)=O)C)CCC(CNC(=O)Cc2cnoc2)CC1 8433,C(=O)(CS(=O)(=O)CCOC)N(CCNC(C(C(CC)C)=O)=O)CCOCCOC 8434,N1(C(CCN(c2ccccc2)CCCCC)=O)CC(NC(c2csnn2)=O)C(O)C1 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8470,C1(C)(NC(Cc2cc(C)on2)=O)CCCN(C(c2cc(C(C)(C)C)oc2C)=O)C1 8471,C1(=CC(=O)NCCOCCOCc2ccccc2)CC2CCC(N2)C1F 8472,N1(C(C)=O)CCc2cc(CCC(=O)C(N3C4CCC3CC4)=O)ccc21 8473,C1(NC(C(C)CO)=O)(CF)CCN(C(=O)COCCCF)C1 8474,N1(C(c2nc(C(=O)OC)oc2)=O)CC2CC2(NC(c2cc(=O)n(C)o2)=O)C1 8475,Cc1ccc2c(=NC3COCCOC3)[nH]c(=NCc3nc(C)c(C)[nH]3)[nH]c2c1 8476,N1(C(C(CCSC)O)=O)CC2CC(N(C)C(c3cccc(CSC)c3)=O)C1C2 8477,C(CCCCC(=O)NC1COCCN(C(=O)Cc2csc(Cl)c2)C1)N(C)C 8478,CC(C)CC(C(=O)NC1CC1NC(c1ccc(Cl)cc1)=O)N(C)C 8479,C1(NC(C2(NC(C)=O)CC2)=O)CC2CCCC(C1)N2C(=O)CCN(C)C.C1CS1 8480,C(=O)(CC(CC(C)C)NC(=O)CC1CC2CC2C1)NCCc1cc(CC)no1 8481,Cc1c(C(N2CCCC2C(=O)NCC(=O)O)=O)c(Cl)nn1C 8482,N1(C(C(CC)=CC)=O)CC(C)(C)OC2(C1)CN(C(=O)C(C(C)C)NC(=O)CO)C2 8483,C(=O)(CP(C)(C)=O)NC(C)CC1CN(C(=O)CCN2CCCC2)C1 8484,N1(C(C2CC(OC)C2)=O)CCOCC1CNC(C1(C(F)F)CCOCC1)=O 8485,N1(C(c2ccnc(Cl)c2)=O)CCC2C(CCCN2C(c2ccc(O)cc2Cl)=O)C1 8486,c1(N(C(=O)NCCOC)C)coc(OCCCCO)n1.c1(O)ccccc1 8487,c1(CN(C(C(=O)NC2CCC(C(=O)OC)C2)C2(C)CC2)C)cc(Br)ccn1 8488,C=CC(CC(=O)NC(COC(F)F)CO)C1CC1 8489,c1(C(=O)Nc2cn[nH]c2)cccc2c1CN(C(=O)CN1C(=O)CSC1=S)CC2 8490,Cc1cc([N+](=O)[O-])cnc1C(=O)NCCNC(c1csc(-c2ccco2)n1)=O 8491,C(=O)(CCCS(C)(=O)=O)NC1(C)CC(NC(C2(O)CC(C)(C)C2)=O)C1 8492,N1(C(C2N(C(c3cc(OC)n[nH]3)=O)CC(F)C2)=O)CCC2(CCN(C)C2)C1 8493,c1(CNC(c2nnnn2C(C)CC)CCOCC)ccc(OC)c(C)c1 8494,Cc1cc(N2CCC(NC(c3cn(CCO)nn3)=O)C2(C)C)ncc1C#N 8495,C1(CC)CN(C)CCN1C(=O)CC(CNC(=O)CS(C)(=O)=O)OC 8496,N1(CC(=C)C)CCCC1CNC(=O)C(C)OC 8497,N1(C(CC(CC)C(C)C)=O)CC(NC(c2csc(C(C)C)n2)=O)C2(CCCC2)C1 8498,C1(C(N2CC3C=CC3C2)=O)(OC)CCN(C(c2csc(C#N)c2)=O)C1 8499,C(=O)(C(C(C)C)n1cnnc1)NCc1cc(C(N2CCC(COC)C2)=O)sc1 8500,c1(NCC2(CNC(=O)CS(=O)(=O)NC3CC3)CC2)nc(Cl)nc2[nH]c(O)nc12 8501,C1(C(=O)NCC2C(CC(=O)NC(C#C)C3CC3)C2)CC2(CCC2)C1 8502,C1(C(=O)NCCCC2(NC(CCCC3C(C)C3)=O)CC2)CC2OC1C1CC21 8503,Cc1cc(C)c(C(N2CCC(C3CC3)C2CNC(=O)CP(C)(C)=O)=O)cc1C 8504,Cn1nc(C(=O)NCC2CCN(C(=O)Cc3ccoc3)C2)c2nc[nH]c(=O)c12 8505,C1(C(=O)NCc2ccc(OC3CCOC3)cc2)CN(C(=O)C2CC2)CCO1.C(CO)O 8506,c1(C(N2CCCC2C(=O)O)=O)cccc(C2(C(=O)O)CCC2)c1 8507,c1(C(=O)NCC(c2cccc(Cl)c2)NC(C=CCCC)=O)ccccc1C1CC1 8508,N1(C(CNS(CC)(=O)=O)=O)CCC(C)(C)C1CNC(C1CC2(C1)CC(O)C2)=O 8509,N1(C(C(C)SC)=O)CCCN(C(c2ccc(CSC(F)F)o2)=O)C(C(C)C)C1 8510,c1(C(N(CCN(C(c2c(C)ncc(C)c2)=O)C(C)C)C)=O)ccc(F)c(F)c1C 8511,N1(CCC(=O)N(C)Cc2ccccc2)CCCCC(NC(=O)CCn2cncn2)C1 8512,CC(C)(C)C(C)(O)C(=O)NCC1(C)CCCN1C(c1cnc2n1CCS2)=O 8513,C(=O)(CC1=NN(C)C(=O)C1)NC1CN(C(C(C)n2ccnc2)=O)CC1C 8514,C(C)(C)(CCCF)NC(CCN(C)C(c1cnc(S)nc1)=O)=O 8515,c1(C(=O)NCC2(c3ccccc3)CC(F)C2)ncc(C(F)(F)F)cc1Cl 8516,CCC(CNC(c1cn(C)nc1SC)=O)(CC)NC(C1CSCC(=O)N1)=O 8517,CC(C)(F)CC(=O)NCc1cccc(CNC(C2CCC(=O)O2)=O)c1 8518,N1(C(=O)C2=COCCC2)CCOC2(C1)CN(C(c1cscn1)=O)C2 8519,S(=O)(=O)(c1ccc(=NCCCCCSC)[nH]c1)NCCN(C(C)C1CC1)OC 8520,CCCC(CNC(=O)CC(C)C)C(=O)N1CC(=O)NC(CC)C1 8521,C(C)(C(=O)NCc1ncnn1CC)(C1CCC1)NC(C(C)OCC#C)=O 8522,C1(NC(CC(CC)OC)=O)CCC2CN(c3nnc(-c4ccon4)s3)CC12 8523,Cc1c(C(=O)NCC2(F)CC(CO)C2)cc(C(F)(F)F)cc1[N+](=O)[O-] 8524,C#Cc1cnc(C(=O)NCc2ccc(C(=O)N(C)Cc3cocn3)s2)c(C)c1 8525,c1(OC)ccc2cc(C(=O)NCC(C)(C(C)C)NC(=O)COC(F)F)[nH]c2c1 8526,C1(NC(c2cn(CC)nn2)=O)C2CC(NC(=O)CC3CCN(C)C3=O)CC12 8527,CCCCCC(O)CC(=O)N1CC2CC1CN2C(C1CCc2nccn2CC1)=O 8528,c1(C2(C(=O)NCC(C)N(C(c3n[nH]c(C)n3)=O)CC)CCC2)ccccc1C 8529,Cc1cc(C2CC2)ccc1C(=O)NCC1CN(C(=O)CCC2(C)CC2)CC1C 8530,C1(NC(c2ccnn2C2CC2)=O)CC(CNC(c2n[nH]cc2)=O)C12CCC2 8531,N1(C(c2cc(C)sn2)=O)CCC(C(C)(C)C)(CNC(C2CC2C#N)=O)C1 8532,N1(C(c2c(C)csc2)=O)CCC2(CCN(C(C3CN4CCN3C(C)C4)=O)C2)C1 8533,c1(C(N2CC3CN(C(CCc4scc(C)c4)=O)C3C2)=O)ccc2ccoc2c1 8534,c1(-c2cccc(CN3C(CO)CSCC3)c2)ccnc2c1CCC2.c1(C)ccccc1 8535,c1(C(=O)NCC(C)CNC(c2ccccc2F)=O)nnn2c1C(=O)NCC2 8536,C1(NS(CCCOCCOC)(=O)=O)Cc2ccccc2C1C 8537,Cc1c(C(N2CCC(N(C(=O)Cc3ccon3)C)C2)=O)c(O)nc2ccccc12 8538,C12(C(N(C3CN(C(C4CC(C)(O)C4)=O)C3)C)=O)CC3CC1C2C3 8539,C(=O)(C(O)CCCNC(=O)CC(C)(C)C)NCC(CC(C)C)OC 8540,C1(CNC(c2c(CC)ocn2)=O)(NC(C2CC(=O)NC(=O)N2)=O)CCCCC1C 8541,C1(C(C)C)CCN(C(C2CC3(C2)CC3F)=O)C(CNC(C2CCOCC2)=O)C1 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8671,S(=O)(=O)(c1ccc2nc(O)oc2c1)N1CCCN(C(C(C)n2cccn2)=O)CC1 8672,C(CCC(C)(C)C)NC(c1c(CNC(C(C)=C(C)C)=O)n[nH]c1)=O 8673,Cc1ccc(C(=O)NC2CC3CC2N(C(=O)CN2CCC(C)CC2)C3)c(O)n1 8674,N1(C(C(C)C2CC2)=O)CCCC2(NC(c3cncc(F)c3)=O)CC2C1 8675,c1(C(C)=O)c(C)[nH]c(C(=O)NCC2(O)CC(NC(=O)CCC3CC3)C2)c1C 8676,N1(C(=O)Nc2cccc(-c3c(Cl)cc(C)c(F)c3)c2)CCc2c(O)noc2C1 8677,c1(C(N2CCC(CC)C2CNC(c2ccco2)=O)=O)cc(F)c(N)cc1F 8678,N1(C(C(C(COCC)C)C)=O)CCc2sc(CNC(=O)COC(C)C)nc2C1 8679,CC1CNCCC1Nc1cccc(C2CC2)n1 8680,c1(CSCC(=O)N(CC(C)NC(CNC(C)=O)=O)C)coc(-c2ccccc2)n1 8681,C1(C(N2C(CN(C(CN(C)C)=O)C)CCC2)=O)CCC(F)(F)CC1 8682,C#CCCCC(C)C(=O)NCC(C(=O)NC1CC(O)C(F)C1)N(C)C 8683,CCCS(=O)(=O)CC(=O)NCCCC(C)NC(=O)CC1(CO)CCOCC1 8684,c1(CN2CCC(CC(=O)Nc3c(OC)ccnc3)C2)ccnc(Cl)c1Cl 8685,C(CCN=c1[nH]c2c(F)cccc2o1)N(C(c1cnoc1-c1cccs1)=O)C1CC1 8686,C1(C(C)=O)CC(CC(N2CCN(C(=O)C(F)=C3CCC3)CC2)=O)C1(C)C 8687,C1(CNC(Cc2c(SC)cccc2)=O)CCC2(CN(C(=O)CC3CN(C)C3)C2)O1 8688,CC(C)(CC(F)(F)F)C(=O)NCC(CO)NC(C1(c2ccsc2)CC1)=O 8689,C1(NC(C(C)(F)F)=O)CC2(C1)CC(CNC(c1cnc(-c3ccc(Cl)s3)s1)=O)C2 8690,N1(C(CCNC(C)=O)=O)CCCC2(C1)CN(C(C1C(C#N)C1(C)C)=O)C2 8691,C12(CNC(c3cc(C)sc3)=O)CCC(CC1)N(C(C1CC1C1CCCO1)=O)C2 8692,C(=O)(CS(=O)C(F)(F)F)N(CC(C)N(C(CNC(C)=O)=O)C)C 8693,C(N=c1[nH]c(=NCCCc2nccs2)[nH]c2cccc(F)c12)c1cc(CC)on1 8694,n1(CC(=O)NCC#CCNC(C2(C)CCOCC2)=O)cnc([N+](=O)[O-])c1 8695,C1(C(=O)NCC2(COC)CN(C(c3ccco3)=O)C2)C2CCCCC12 8696,C1(C(N2CCC(C)(NC(Cc3cc(OCC)no3)=O)C2)=O)CC(C)CC(C)C1 8697,N1(C(COCCCC(C)C)=O)Cc2nccn2CC(NC(=O)C2CC2)C1 8698,C12(CNC(C(C)Nc3ccc(Cl)cc3)=O)CC(NC(=O)C(N)=O)(C1)C(C)O2 8699,C(=O)(C1CCc2c[nH]nc21)NC1CC2CN(C(c3n(CC)nnc3)=O)CC21 8700,N1(C(C#CC(C)C)=O)CC2COCCC2(NC(c2ccc3nc(S)[nH]c3c2)=O)C1 8701,C1(NC(C2(C)CCOC2)=O)CC12CCN(C(c1ccc(S(C)(=O)=O)o1)=O)CC2 8702,Cc1cc(C(N2CC(F)CC2C(N2C3CCC2CC(O)C3)=O)=O)c(F)cc1F 8703,N1(C(C=C(CCC)C)=O)CCN(C(=O)CSc2ccc(Cl)cc2)C(C)CC1C 8704,C(C(=O)N=c1ccn(CCC)[nH]1)c1nccc(CNC(CCCCC=CC)=O)c1 8705,N1(C(c2c(CC)cccn2)=O)CCN(C(c2cccc(N)c2C(F)F)=O)CC1C 8706,C1(C(N(C2CCC2)CC#C)=O)CC2CCC(C1)N2C(=O)Cc1ccon1 8707,c1(C(=O)NCC(CC=C)NC(=O)Cn2ccnc2CCC)nc(C)ccc1OC 8708,c1(C(N2C(CC=C)(C(=O)NCC3(CCC)CC3)CCC2)=O)cnn(C)c(=O)c1 8709,CC1=C(C(=O)NCC2CCCCN2C(c2cccc3nonc23)=O)CCCC1 8710,c1(CCC)nnc(S)n1CC(=O)NC1CCC(NC(C2CCN(C)C2C)=O)CC1 8711,C1(CC(=O)N(CCNC(C(C)(C)NC(=O)OC)=O)CC2CC2)CCCCCC1 8712,C#CCCCCCC(=O)NCC1(CNC(C2CC2=C)=O)CC1(F)F 8713,C12(NC(C3CC(=O)NC3)=O)CCC(C(=O)Nc3nccnc3CO)(CC1)CC2 8714,c1(C(N2CCC(NC(C(C=CCCC)O)=O)C(O)C2)=O)cnc2n1CCOC2 8715,O=S(=O)(c1ccc2c(c1)CC2)NC1(c2cccc(OC(F)F)c2)CC1 8716,N1(C(c2c(CC)cco2)=O)CC(NC(c2cncc(F)c2)=O)C(C(F)(F)F)C1 8717,c1(CN2C(C(N(C3CC3)CC)=O)CC3(CC3)C2)cc(OC)c(O)c(Br)c1 8718,c1(OC)ccc(C(=O)NC(C)CC(C)NC(c2cncnc2)=O)cc1C(F)F 8719,N1(C(C(C)=C(CC)C)=O)CCC2(NC(C3CS(=O)(=O)C3)=O)CCCCCC12 8720,N1C(NCc2c(COC)nccc2)=NCCOCC1.C(C)(C)(C)OC(=O)N(C)C 8721,C1(NCc2[nH]c(=N)sc2)CCCCC1C(=O)NCc1ccccc1N1CCCC1 8722,N1(C(=O)NCCC(=O)OCC)CCC2CN(C(=O)Nc3ccc(F)c(Cl)c3)CC12 8723,C12(NC(C3N(CC)CC3)=O)CC(C1)N(C(=O)CCn1cc(Cl)cn1)C2 8724,C1(NC(c2ccc(SC)s2)=O)CC2CC(NC(=O)C=Cc3cc[nH]n3)CC2C1 8725,c1(-n2cc(C(N(C(C)CCNC(C3CC(C#N)C3)=O)C)=O)nn2)ccccc1Cl 8726,c1(OC)cnc(C(N2CCCCC2CCCNC(=O)Cc2c[nH]nc2C)=O)cn1 8727,C1(NC(c2cnsn2)=O)CN(C(c2sccc2OCC(F)(F)F)=O)CCC1CO 8728,C1(C2CCCN(C(C3CC(F)C3)=O)C2)(NC(C(C)NC(=O)CC(C)(C)C)=O)CC1 8729,c1(C(=O)NC(CC(C)NC(c2occ(C)c2C)=O)C)ccc(=NCC2CC2)[nH]c1 8730,c1(OCCN(C)C)ccccc1C(=O)NC1C2CC1N(C(=O)CN1CCSCC1)C2 8731,c1(OC(C)(C)C)ccc(CNC(=O)CN2CCC(=O)NC2=O)c(O)c1 8732,C=C1CCC(C(N2CCCCC2C(=O)NC(C)C)=O)CC1 8733,C1(OC)CC(SCCCOCCC(=O)OCc2cccs2)C1 8734,C1(NC(c2ccc(OCCN)c(F)c2)C)CC2CCC(C1)O2.C(C)(C)(C)O 8735,N1(C(C23N(C(C4(CC)COC4)=O)CC(C)(C2)C3)=O)CCC2(CC1)CSC2 8736,c1(OCC(=O)NCC2CC(CNC(=O)CCF)CO2)ccc2c(c1)CCCC2 8737,N1(C(CC(C)(C)n2cc(C(C)Sc3nncs3)nn2)=O)Cc2ccccc2C1 8738,c1(OC)cc(C(=O)NCCC(O)CNC(=O)C(C)(C)C)ccc1[N+](=O)[O-] 8739,C(=O)(C1=CS(=O)CCC1)N1CC(C=O)C1.c1(C=O)cocn1.CCO 8740,CC(N=c1cccc(S(=O)(=O)NCC23CCCC2C3)[nH]1)C1CCOCC1 8741,C1(O)(CN(C(C(F)=C(C)C)=O)C)CCN(C(=O)C(C(C)(C)C)C2CCCC2)CC1 8742,N1(C(c2ccc(Br)cc2)C(=O)NCCSC)CCc2cc(F)cc(F)c2C1 8743,N1(C(C2(CCCC)CC2)=O)CCN(C(=O)C(O)C2CC2)CC2(CC2)C1 8744,C(CN=c1[nH]c2c(c(=NC(C)c3cncc(F)c3)[nH]1)CCC2)(C1CCCC1)OC 8745,c1(C(=O)NCC23CN(C(c4n(C)nnc4)=O)C(CC2)C3)c(S(C)(=O)=O)cnn1C 8746,N1(C(C2CC(C)(CNC(CCNC(C)=O)=O)C2)=O)CCS(=O)(=O)CC1 8747,c1(CCC)noc(CCC(=O)NC2CCCC2NC(C2CC2C)=O)n1 8748,N1(C(C=C2CCN(C)C2)=O)CC2CC(C1)CN(C(C1CC(=O)N(C3CC3)C1)=O)C2 8749,C(N=c1nc2ncn(C)c2c(NCC2(C)CC(C)C2)[nH]1)c1nn(CC)nc1C 8750,c1(C(=O)OCc2c(NC(CC(COC)C)=O)cccc2)cn(C)c(C)cc1=O 8751,c1(C(N(C(C)CN(C)C(C2CCOC2)=O)C)=O)cc2c(nn1)OCCS2 8752,c1(C(N2CCC(NC(=O)CC3(CO)CC3)C2)=O)cc(-n2ccnc2)ccn1 8753,c1(C(N2CCN(C(COCC)=O)C(CO)C2)=O)cc2cc(Br)ccc2c(=O)o1 8754,C1(C(=O)NC2(CCC)CCC2)CCCN(C(=O)Cn2cc(C#N)cn2)C1CC 8755,c1(CNC(CSCCC)=O)ncoc1C1CCN1C(=O)CCOC(C)CC(C)C 8756,C1(NC(=O)CN2CC=CC2)COC2(CCN(C(C3CC34CCSCC4)=O)CC2)C1 8757,CC(CC(F)(F)F)C(=O)NCCCCN(C)C(C1(C)CCNC1=O)=O 8758,Cc1ccc(F)c(C(=O)NCC(C)CN(C)C(C23CCC(C2)OC3C)=O)c1 8759,c1(C(=O)NC2C(NC(c3nc(CCC)oc3)=O)CC2)ccc(NC(C)=O)cc1Cl 8760,c1(OC)ccc(C(N2CCN(C(=O)C(C)(C)OC3CCC(OC)C3)CC2)=O)cc1 8761,Cc1nc(O)c(Br)cc1C(=O)NCCCNC(=O)Cc1ccc(O)nc1 8762,C(=O)(C(F)(CC)C(=O)OC)NC1(CNC(c2c(CC)occ2C)=O)CCOC1 8763,c1(CC)ccc(C(=O)NCC(C(C)C)NC(=O)C(c2cnccn2)C)c(Cl)c1 8764,N1(C(c2nc(CC)sc2)C(=O)NCc2nnn(C)n2)CCOC(C2(C)N=N2)C1 8765,CCCCC(CNC(=O)C(C1CCOC1)OC)NC(=O)CSC(C)(C)C 8766,N1(C(C2CC(SC)C2)=O)CC=C(CNC(=O)CCNC(=O)CC(C)C)CC1 8767,c1(NC2CCN(C(C=CCC)=O)CC2C)c(Cl)cccc1[N+](=O)[O-] 8768,c1(N2CCCC(COC)C2)nc(=N)[nH]c(=NCC(=O)N(CCCN(C)C)C)[nH]1 8769,Cc1sncc1C(=O)NC(C)CCNC(=O)CC1(C)CC1 8770,N1(C(CC2C=CC(NC(C3CN(CC)C(=O)C3)=O)C2)=O)CC2(C1)NC(=O)NC2=O 8771,N1(C(c2c(C)oc(CO)c2)=O)CCN(C(c2ccc(N=[N+]=[N-])cc2)=O)CCC1C 8772,c1(N2CC(C(C)C)NC(=O)C2)nc(=NCC(C)C(C)(C)C)[nH]c2c1CSC2 8773,Cc1nnccc1C(N1CC2CC1C2C(=O)NCCc1ccncc1)=O 8774,c1(C(=O)NC2CC(CNC(=O)C3=COCCO3)CC2O)nsc2c(Cl)cccc12 8775,C12COCCN1C2=O.C1(C)(C(C)C)CC1C(=O)NCC12CC(C1)C2 8776,c1(CC(=O)NC(C2CCCN(C(C(C(C)C)NC=O)=O)C2)C)ccc(Cl)cc1F 8777,c1(NCCCN(c2ccccc2Cl)CC)cc(Cl)nn(C)c1=O 8778,Cc1ccnc(C(=O)NC2(C3CCCN3C(=O)CC3CCCC3O)CC2)c1 8779,C(=O)(C1=NNC(=O)CC1)Nc1ncc(CCNCCn2c(C)ncc2)s1 8780,N1(C(c2ncc(I)s2)C(=O)NC(CC)C)CCC(c2ccnn2C)CC1 8781,CCC(CC(F)F)C(=O)NC1CCCCC1NC(c1c[nH]cc(Br)c1=N)=O 8782,CC(O)CCCCCC(=O)NC1CN(C(c2cnn(CC3CCOC3)c2)=O)C1 8783,CC(C)CCC(N)C(=O)NCC(c1ccco1)N1CCCC1 8784,C#CCCC(O)C(=O)N1CCCCC1CNC(c1cnccc1C)=O 8785,C1(NC(C(C(C)C)=O)=O)CN(Cc2ccc(C(N)=O)cc2)CCC1(F)F 8786,C1(C(N(CC(C)(C)NC(c2c(CC)nco2)=O)C)=O)CCCCC1(F)F 8787,C1(CNC(=O)Cn2cnnn2)CN(C(c2cccc(-c3nc[nH]n3)c2)=O)CCO1 8788,C(=O)(CC1=CCCC1)NCC(CC)NC(c1ccccc1C(=O)NC(C)(C)C)=O 8789,C1(CC)(CNC(C2OCCC2CNC(=O)CC2(OC)CC2)=O)CCCO1 8790,CC(C)(C)C(O)CC(=O)N1CC(CNC(c2ccc(C(F)(F)F)[nH]2)=O)C1 8791,C(=O)(C1Cc2c(Cl)cccc21)N(C1CCCN(C(c2nnc(CC)o2)C)CC1)C 8792,C1(N(C)C(C2CC(C)(F)C2)=O)CCCN(C(=O)CCc2ccc(Cl)cc2)CC1 8793,CN1CCCCC1CC(N1CC(C(=O)NOCCc2ccccc2)(CF)C1)=O 8794,C1(NC(NCc2cc(C)on2)=NCc2ccccc2C2CC2)CC(C)OC(C)C1 8795,c1(C(N2CCC(N(C(=O)CC(=O)N(C)C)CCC)C2)=O)c(Cl)ccc(O)c1Cl 8796,Cc1cc(F)ccc1CC(=O)NCCC(C)N(C)C(c1cccc(F)c1O)=O 8797,Cc1ccn(C(C)(C)C(=O)NC2(C)CC(NC(=O)CSC3CCCCO3)C2)n1 8798,c1(N)nc(C)ccc1OC.C1(C)(CC(=O)N(CCC)CCNC(=O)COC)CCCC1 8799,c1(CC(N2C(CNC(C3C(CC)OCC3)=O)CC2)=O)cccc(F)c1O 8800,Cc1cnc(NCc2c(C)cccc2C)c(S(=O)(=O)N2CCC(C3CCC3)C2)c1 8801,C1(C(N(C)CC2CN(C)C2)=O)CN(C(=O)C(C2(O)CCCC2)F)CCO1 8802,c1(CC)nn[nH]c1C(=O)N(C)CCNC(C1(COC)CCOC1)=O 8803,C1(C(=O)NC(C(N2CCCC(OCC)C2)=O)C)CCC2(CCC2)C1 8804,N1(C(CC=CC=C)=O)CC(CCCC)C(C)C1.c1(CNCC)cnc(CC)[nH]1 8805,C(=O)(C1SCCc2ccccc21)N1CC(C(C)NC(=O)CC2(C)CC2)C1 8806,C1(N(C(=O)CCCCC2CC2)C)CCCN(C(c2cccc(F)c2N)=O)CC1 8807,c1(C(N2CC3C(CNC(C(C)c4cccs4)=O)C3C2)=O)coc2cccc(O)c12 8808,c1(C(N2CCCC3(NC(C=CCCC)=O)C(C2)C3)=O)cc2c(cc1O)CCCC2 8809,CC(C)C(O)C(C)C(=O)NCC12CC1CN(C(=O)CCc1ccccc1)C2 8810,CN1CCNNS(=O)(=O)c2cc(N=c3[nH]c4ccccc4s3)ccc21 8811,c1(C(N(CC(=O)N(C(C(N)=O)C2CC2)C)CCC)=O)ccc(N)cn1 8812,C1(C(N(CCCNC(=O)CC2(OC)CC2)CC)=O)(OC)CCCOC1 8813,N1(CCN(C(=O)CCN2CCOCC2)C)CCN(C(C2(C)CCCC2O)=O)CC1 8814,c1(-c2cn(CC3N(C(C(C=C)CC)=O)CC3)nn2)cc(N)cc(F)c1 8815,Cc1ncc(NC(C2CC(C)(NC(=O)CC3COCCO3)C2)=O)c(C)c1C 8816,c1(CC(=O)NC2C(C)CN(C(=O)C3=CCSC3)C2)cccc2cnccc12 8817,c1(C(=O)NCCOCCOCCNC(C2(O)CCOC2)=O)ccc2c(c1)CCO2 8818,C1(C(N2CCC(NC(Cn3cc(C(=O)OC)nc3)=O)C2)=O)CC2CCC1O2 8819,c1(C(=O)NCCC(CNC(COCCSC)=O)O)cccc2ccn(C)c12 8820,N1(C(c2c(C)cno2)=O)CCCCC(CNC(=O)Cc2cn(C)nc2C)C1 8821,c1(NCc2c(C(=O)Nc3c(C)cnc(Cl)c3)cccn2)ccc2ncccc2c1 8822,C(=O)(C(O)CCC(F)(F)F)NCC1C(NC(C2(OC)CCC2)=O)CCC1 8823,C1(C(=O)NC(c2c(C)cccn2)C)CC2(CC(NC(=O)Cn3nccn3)C2)C1 8824,C(CCF)(C(=O)NCC1(C)CCCO1)NC(CCCOCCC)=O 8825,Cc1nc(CCNC(c2cc(Cl)cc3cc[nH]c23)=O)nc2c1CCC2 8826,C1(CC)CCCN(C(=O)CC(C)(C)C2CC2)C1C(N1CC2(CC2)CC1CO)=O 8827,Cc1onc(CO)c1C(=O)NCC1CCN1C(C1CC(C)(CN2CCCC2)C1)=O 8828,C1(CC(=O)NC2CN(C(c3ccc(SC)s3)=O)CC2C)CCC2(CCCC2)CC1 8829,C1(C(=O)NC(C)C)CCCC(C(=O)Nc2cc(C3CCOCC3)nn2C)C1 8830,C(=O)(C1Cc2c(Cl)cccc21)NCCN(C)C(c1cnc(CCC(F)(F)F)s1)=O 8831,c1(C(=O)NC2C(NC(C(CCSC)N(C)C)=O)COCC2)ccnc2[nH]ncc12 8832,c1(C(N(CCC)CCNC(C2CC2(F)Cl)=O)=O)nc(C)c(C)nc1C 8833,N1(C(C(C)(C)C2CCCO2)=O)CCC(O)(CNC(=O)CC2CSC2)C1 8834,CC(C)CC(C)(CO)NC(=O)C(C)C(C)NC(c1c[nH]nc1C(C)C)=O 8835,N1(C(c2n(C)nnc2)=O)CCN(C(=O)CN2CCOCC2)CC1c1ccccc1 8836,N1(C(C=C(C(=O)N(CCC)CCC)F)=O)CCC(C)C1CSC 8837,c1(C(N(CCCC(=O)NC2CCSCC2)C)=O)ccc2[nH]nc(Cl)c2c1 8838,N1(C(N)=O)CCC(NC)CC1.N12CCCCC1c1nnc(o1)CS2(=O)=O 8839,c1(C(C(=O)NCCSC)N(c2cc(Cl)no2)Cc2ccccc2)cc(I)cn1C 8840,c1(C(C(=O)NC(C)(C)CC)N(C(C#C)C2CCC2)C)cnc(C)nc1 8841,C12(C(N)=O)CCCC1(C(=O)NCCOCCCNC(=O)CC1(O)CCC1)C2 8842,N1(Cc2cccc(C(=O)NCC(C)C#N)c2)C(=O)CN(C)C1=O 8843,c1(C(=O)NC(CC(=O)NCC=C)CC2CC2)cccc(C)c1F 8844,c1(C(N2CCC(NC(c3cnc(C)nc3)=O)C2C)=O)cc2c(Cl)cccc2[nH]1 8845,C1(C(N2CCC(NC(CC(C)n3cccc3)=O)CC2)=O)CC2CCC(C1)C2F 8846,C(C(=O)NOCC1CC1)C(C)(C)CNC(C1COCC1C(N)=O)=O 8847,C(C1C(C(=O)NCC2CCCCN2C(=O)C(C2(O)CCCC2)F)C1(C)C)=C(C)C 8848,C(=O)(CC(C)CC(=O)OC)N1CCC(CC=C)(NC(=O)C#CC(C)(C)C)C1 8849,n1(CCC)ccnc1C(F)(F)C(=O)NC1CC(C(C)NC(=O)C(F)CSCC)C1 8850,c1(C(=O)NC2(C)CC(NC(COCCN(C)C)=O)C2)cc(O)nc(Cl)c1 8851,C(C(=O)N1OC2CCC1CC2)(N(C)C(c1c[nH]nc1Cl)=O)C1CC1 8852,Cc1cccc(F)c1C(=O)NCC1CC1NC(=O)C(C)(C)NS(C)(=O)=O.C(N)=O 8853,C1(O)(C(=O)NCC=C=C)CCN(CC(C)CO)CC1 8854,c1(NCc2scc(CC)c2)ccc(SC)cc1.C1(C)C(=O)N1C(C)C 8855,C(=O)(C(F)CC(C)(C)NC(c1ncccc1O)=O)NCC(CC)(C)Cl 8856,C1(C(N2CCN(C(C)=O)CC2c2cnn(C)c2)=O)CCc2cnc(C)n2C1 8857,C(=O)(C1=Cc2ccccc2C1)NCC1(C)CN(C(c2cnc(O)s2)=O)CCO1 8858,C1(C(=O)NCCCN(CC)CC)C=CCC(NC(c2cnn(CCO)c2)=O)C1 8859,c1(C(=O)NC2CN(C(C=COCC)=O)CC(O)C2)[nH]c2c(c1C)CCCC2 8860,C=CC(C)(C)CC(=O)N1CCN(C(c2[nH]ccc2C2CC2)=O)CC1CF 8861,c1(C(=O)NCCCN(C(COCC(=O)NC)=O)C(C)C)cscc1SC 8862,C1(CN(C)C(c2cnn(C(C)(C)C)c2)=O)COCCN1C(=O)CC(Cl)Cl 8863,Cc1cc(C(=O)NCCNC(c2cc(C(=O)C(C)C)c[nH]2)=O)nn1C1CC1 8864,c1(N(CCN(C(C)C)C(c2ccncc2Cl)=O)C)ncc2c(Br)cccc2n1 8865,N#Cc1ccc(C(N2CCSC3CCC23)=O)cc1O 8866,C(=O)(C(CC(C)C)SC)N1CCC(C(=O)NCC(C(=O)OC)(F)F)(NC(C)=O)C1 8867,c1(C(N2C(C(=O)NCC34CC(CCO3)C4)CC2)=O)coc2ccccc12 8868,n1(CC)ccc(C(=O)NCC2(F)CCN(C(=O)C(c3ccnn3C)O)C2)cc1=O 8869,Cc1cc(C(N2CCCCC2C2(NC(=O)CC(C)F)CC2)=O)cc([N+](=O)[O-])c1Cl 8870,c1(C(N2C(C)CC(CNC(C=C(CC)C)=O)C2)=O)ccc2c(c1)C(=O)NCC2 8871,Cc1nc(CC(N2CC(C)(C(=O)NC3CONC3=O)C2)=O)co1 8872,C(=O)(C1CSc2ccccc21)NC1CCC(CNC(c2ncncc2F)=O)CC1 8873,c1(C(CNC(c2cnc(CC)s2)=O)NC(C2CCN(C)C2)=O)ccc(F)cc1F 8874,n1(CCOC)ccc(=NC(=O)C2C(CNC(c3[nH]ccc3C)=O)C2(C)C)[nH]1 8875,NS(=O)(=O)c1cnn(CC(N2CCCCC(NC(=O)C=CC3CC3)C2)=O)c1 8876,N1(CCC)CCN(Cc2n[nH]c(CC(=O)O)n2)CC1C.C12CN(C1)C2=O 8877,C1(CNC(CCOCC)=O)COCCN1C(C1CCSC1)=O 8878,n1(CC)nnc(C(N2CCC2CNC(=O)CNc2nccs2)=O)c1C 8879,c1(N(C(CNc2ccc(Oc3ccccc3)cc2)=O)SC)c(C)cccc1C#N 8880,C(=O)(C(CC)C(=O)N1CC(C(=O)NCC2CC3(CC(OC)C3)C2)(OC)C1)OCC 8881,CC1CN(C(=O)CCCC#N)CC(C)N(C(c2cc3sccc3[nH]2)=O)C1 8882,C1(O)(CNC(C2OCCN(C(C)C)C2)=O)CCCNCC1 8883,CN1CCN(C(C2C=CC=CC=C2)=O)CC1C(N1CCC2CC12)=O 8884,C(=O)(CCCCC(C)C)N1C(CNC(c2c(C)cco2)=O)CCC1 8885,C1(NC(CCC(CC)OC)=O)(CNC(C2CCCN2N=O)=O)CCC(F)(F)CC1 8886,c1(C(N2CCN(C(c3[nH]cc(C#N)c3)=O)CC2CCO)=O)nccc2nn[nH]c12 8887,c1(C(=O)NC2C(CNC(c3c(C)nns3)=O)CCC2)ccc(F)c(F)c1N 8888,C1(NC(c2c(CCC)n(CC)nn2)=O)CCCN(C(c2conc2C)=O)CC1 8889,C1(NC(C(C)Cc2ccc(F)cc2)=O)CC2CC(NC(c3ccsc3)=O)C2C1 8890,C1(CNC(C(CC=C)CC)=O)CN(C(=O)CCC(=O)OCC)C2COCC2O1 8891,C1(NC(CC(C)C)=O)CCCC(NC(=O)CC2CCC(=O)C2C)C1 8892,c1(-c2scc(CN3CCN(CCCCC)CC3)n2)ccc(F)c(OC)c1 8893,c1(C(N2C(C(=O)NC3CONC3=O)CSCC2)=O)ccc2sccc2c1O 8894,C1(CC)C(NC(C2CC2C(=O)OCC)=O)CCCN1C(C1CC(C)(C)CN1C)=O 8895,C1(CC=C)N(C(c2cccc3c2CCO3)C(=O)NCCSC)CCCC1(C)C 8896,C1(C(N(CC(=O)NC2CCC2)CC2CC2)=O)CCCC1.C1(CC#C)CC1 8897,C1(C(=O)NC(C)C2CC2)CCN(C(=O)C2=NOCC2)C(C)(C)C1 8898,c1(C(N2CC(OC)(CNC(=O)CC3CCOC3C)C2)=O)c[nH]nc1[N+](=O)[O-] 8899,c1(C(CCC)C)nc(-c2cc(COC)ns2)n(-c2cncc(Br)c2)n1 8900,N1(C(C(C)=C(CC)C)=O)CC(C(=O)NCCC2(C)CC2(F)F)C(C(C)C)C1 8901,C1(NC(NCc2sccc2)=NCC2CCCO2)CCCC12CCC2 8902,C(C(C)(C)C#CC(=O)NC(C)CN(C)C(C)C)OC.c12ccc(cc1)CC(=O)N2 8903,O=C1OC(C(=O)NCC2CCN2C(=O)Cc2cn[nH]c2)Cc2ccc(Cl)cc21 8904,Cc1ccc(C)c(CC(=O)N(C(CNC(c2cncc(C)c2C)=O)C2CC2)C)c1 8905,c1(NC2C(OCC)CCCC2)c(CSC2CCN(C)CC2)oc2ccccc12 8906,N1(C(CSCC(N)=O)=O)CC(S(=O)(=O)N2CCN(C(C3CCCSS3)=O)CC2)C1 8907,C1(CCCC(=O)NCC(CNC(c2n(C)ccn2)=O)CO)CCCC(=O)N1 8908,S(=O)(=O)(c1ccc([N+](=O)[O-])cc1OC)N1CC(C(=O)OC)C(N)C1 8909,C(C(C(C)(C)C)NC(c1c[nH]nc1C1CCCO1)=O)NC(C=CCOC)=O 8910,c1(CCC(=O)N(CC(C)NC(C2CC2(Br)Br)=O)C)cncnc1 8911,c1(CC(=O)NCC2CNCCOC2)ccc(Br)c(O)c1 8912,N1(C(C2C(OCC)CC2)=O)CCC(CNC(=O)C(CN(C)C)CC)C(C)(C)C1 8913,C(=O)(C(CO)C(F)(F)F)N(CC(C(N1C2(CC(COC)C2)CC1)=O)C)C 8914,N1(C(CCN(CCOCCOC)C)=O)CCC(CC)C1CNC(c1ccc[nH]1)=O 8915,CCCC(C(=O)NCCn1cc(C(N2CCC(N3CCC3)CC2)=O)cn1)OC 8916,N1(C(c2c(CCC)cccc2)=O)CCC2(CCCCN(C(=O)C3CCCS3)C2)C1 8917,N1(C(c2cc(CC)nc(O)c2)=O)CC2CN(C(=O)CN(C)S(N)(=O)=O)CC2C1 8918,C1(CC(=O)N(C)CCNC(=O)CC2(C)CCC2)COCC1(C)C 8919,C1(C(=O)NC)CCN(C(=O)C(C)N(C)C)C1C.c12cnn(c1)CCNC2=O 8920,Cc1nnc2c(C(N3CCC(CNC(C4CCC4)=O)C34CCC4)=O)cccn12 8921,CC(C)(CCC(=O)N1CC(NC(c2ccc(Cl)c(Cl)c2O)=O)C1)[N+](=O)[O-] 8922,C=CCCCC(=O)NC(CC1CC1)C(=O)NC1CCCC1 8923,C1(O)(Cn2cc(C(C(C)C3CC3)NC(C(CC)OCC)=O)nn2)CCCN(C)C1 8924,C(c1c(F)ccc(Cl)c1F)=CC(N1CC2C(NC(CC(C)C(F)F)=O)(C2)C1)=O 8925,c1(C(=O)NCC(CO)NC(C=CC=CCC)=O)cc(S(N)(=O)=O)c(C)o1 8926,N1(C(CCCC(CC)CC)=O)CCOC2(CCN(C(=O)CSC(F)F)CC2)C1 8927,C(=O)(CC(=O)NCc1nc[nH]n1)NC(C1(C(=O)NCC(F)F)CC1)C 8928,Cc1cncc(C(N2CC(NC(C3CNC(=O)N3C)=O)C(C)C2)=O)c1 8929,N1(C(C(CCC)C)=O)CCN(C(c2n[nH]c(C)c2F)=O)C(CC(C)(C)C)C1 8930,C(=O)(C1CCCn2ncnc21)N1C(C(=O)NC2CN(C(C)=O)C2)CC2COCC21 8931,N1(C(C2CC(C)=C(C)CC2)=O)CCC(C)N(C(=O)C(c2cnn(C)c2)C)CC1 8932,C1(CC(=O)N(CC(CC)NC(c2c(C)ncnc2C)=O)CC)CCC(F)(F)CO1 8933,C1(N(CCC)C(C2CC2C2CC2)=O)CCN(C(c2ncn(C)c2C)=O)CC1 8934,c1(CNC(C2CCN2C(C2(F)CCCC2)=O)=O)cnccc1Cl 8935,C1(O)(CNC(c2c(CNC(CC=C=C)=O)n[nH]c2)=O)CCCOC1 8936,C1(F)(C(=O)NC2CC(OCC)C2)CCN(C(c2sc(C)nc2C(F)(F)F)=O)C1 8937,C(C1CCOCC1)=CC(=O)N(C(C)C(=O)Nc1cnn(CC)c1C)CC 8938,C1(C)(C(=O)NCC2CN(C(c3c(CC)occ3)=O)CC2O)CCCCC1(F)F 8939,C1(CC(N2CC(C)(NC(C(C)OCCOC)=O)C2)=O)COc2ccccc2O1 8940,CC(C)(C)C(C)(C)C(=O)N1CCC(C)(NC(=O)Cc2cccc(O)c2)C1 8941,CC(C)CC(CNC(=O)CC1CCC(C(F)(F)F)O1)NC(C1(C)CCOCC1)=O 8942,c1(C(N(C)CC2OCCN(C(c3cc(C)c(C)o3)=O)C2)=O)cccc(=S)n1O 8943,N1(C(C2C(OC)CCC2)=O)CC2CCC1CN2C(C1(CO)CC(C)(C)C1)=O 8944,c1(C(=O)NC2COCC2NC(C2CCCOC2)=O)ccnnc1S 8945,N1(C(c2nc(CCCC)sc2)=O)CC2CCC1C(CNC(=O)C(CO)N(C)C)C2 8946,C1(O)(CCNC(C(C)C2CCOC2)=O)CCN(C(c2coc(C(F)F)c2)=O)CC1 8947,C1(C(N(CC=CC(NOCC2CC(=C)C2)=O)C)=O)C2CCC(C2)C1C 8948,c1(C(=O)NCCNC(CC2(C#N)CCCCC2)=O)ccc(S(=O)(=O)CF)cc1 8949,C1(CC(=O)NCCCCCN(CC)CC)CN(C(=O)C(C)OC)CC1C 8950,N1(C(CC2(C(F)(F)F)CC(=O)NC2)=O)CCn2cccc2C1CC 8951,N1(C(C(n2cc(Cl)cn2)C)=O)CCC(CCNC(C2CN(C3COC3)C2)=O)C1 8952,c1(C(=O)NCCC2N(C(Cc3cnc(C)s3)=O)CCC2)ccccc1F 8953,C1(COC(=O)NCC(C(=O)OCc2ccccc2)C2CC2)CCC(C2CC2)CC1 8954,N1(C(c2cnc(Cl)s2)=O)CCCC(NC(=O)CSCc2ccc(F)cc2)C1 8955,c1(C(=O)NCC(CN(C)C(c2c(Cl)cccc2Cl)=O)O)coc2c1C(O)CCC2 8956,c1(C(=O)NC2CC3(CN(C(C4(N=[N+]=[N-])CC4)=O)C3)OC2)cc(Cl)cc2c1CCC2 8957,c1(C(N(CCCC(=O)OC)C(=O)CCNC(C)(C)C)C)c(Cl)cnn1C 8958,CCC(CC(F)F)C(=O)N1CCC(NC(c2cc3ccccc3s2)=O)C1C 8959,c1(CN(CC(=O)N(CCCOC)C)C(=O)COC)cnncc1O 8960,N1(C(C2(C#N)C(C)C2)=O)CCC2(CC1)CN(C(=O)CCNC(=O)C=CCl)C2 8961,C(CC)(C(C)(F)F)NC(CC(C)N(C(CCSCCCC)=O)C)=O 8962,C(CC(O)C(F)(F)F)NC(C(CCN(C)C)NC(C=CCOC)=O)=O 8963,c1(N2CCC(OC)C2)ccc(S(=O)(=O)NCC(O)CC2CCC2)c(Cl)c1 8964,C1(C(=O)NCC2(NC(C(C)C3CCOC3)=O)CC2)CC(=O)c2ccccc2O1 8965,C1(NC(CC(C)n2ccnc2)=O)CC12CC(NC(C13CC(C)(C1)C3)=O)C2 8966,c1(CNC(C2CC23CN(Cc2ccnc(Cl)c2)C3)=O)cc(Br)ccc1O 8967,C1(C(N2CC(NC(c3n[nH]c(CC)c3Cl)=O)C3(C2)CC3)=O)CC=C(C(C)C)CC1 8968,CCC(C)(COC)C(=O)NC1CC2C(NC(=O)CCc3ccnc(C)c3)C2C1 8969,c1(C(=O)NCC2CCC(NC(C(CC)OCC)=O)C2)c(C)c(C)cc(C)c1C 8970,N1(C(CSCC#C)=O)CCC(CCNC(C2CCCCO2)=O)C1 8971,C1(CC=C)(NC(=O)Cc2ccco2)CCN(C(=O)C(F)OC(F)(F)F)C1 8972,N1(C(C2N(C(CNC(=O)OCC)=O)CCC2)=O)CC2CCCC2(CO)C1 8973,N1(C(C2C(OCC)CC2)=O)CC2CCC(C1)N2C(=O)CCc1ccon1 8974,Cc1cc(=O)ccn1CC(=O)NCC1(C(C)NC(c2ccncc2)=O)CC1 8975,C(C)(CCCCCO)NC(C(CSC)(C)NC(C1CC=CCC1)=O)=O 8976,C12(C(=O)NC3C(NC(C=C(C)c4cccs4)=O)CCC3)CCN(CC1)S(=O)(=O)C2 8977,N1(C(c2c(OC)cncc2)=O)CC2CC(NC(C3CCN(C)C3)=O)CC1C2 8978,C(=O)(CCCC(=O)C(C)SCC(c1ccccc1C(F)(F)F)(C)OC)OC 8979,CCC(C)C(C(=O)N1CC(CC(=O)NC2CCOCC2F)(OC)C1)N(C)C 8980,Cc1[nH][nH]c(=NC(=O)c2cc(Cl)ncc2NCc2cc(Br)ccc2[N+](=O)[O-])c1C 8981,N1(C(C(C)n2cnnn2)=O)CCC2(CCC2CNC(C2CC(C#N)C2)=O)CC1 8982,CC1(C)CC(CNC(=O)CNC(=O)OC(C)(C)C)CN1C(=O)CCS(N)(=O)=O 8983,c1(C(CC)NC(=O)NCc2ccc(Cl)nc2C)cccc(S(N)(=O)=O)c1 8984,C1(NC(c2ncn(CC)n2)=O)COCCC1C(=O)N(CCO)CCO 8985,c1(C(=O)NCC2(F)CC(NC(c3cnns3)=O)C2)ccc([N+](=O)[O-])cn1 8986,N1(C(C(=O)NCC)=O)CC(OC)CC1(C)CNC(C1(C#N)CCSCC1)=O 8987,CC1CCN(C(C2CC23CCSCC3)=O)CC1NC(C1CN2CCN1CC2)=O 8988,CC(F)(F)CC(=O)NCC1CC1CNC(c1cnc(Cl)[nH]1)=O 8989,C1(C(N2CCC(C)CC2)=O)CC(O)CCN1Cc1cnc(-c2ccccc2)s1 8990,CC(CO)(CO)C(=O)NC1CC1C(=O)Nc1ccccc1OC(F)F 8991,c1(OC)cccc(C(N2CC3C(NC(=O)Cn4ccnn4)C3C2)=O)c1Br 8992,C(=O)(C(C)CC(=O)N(CCC(N1CC(N=[N+]=[N-])C1)=O)C)OC 8993,C1(CC(=O)NC2C(CC)N(C(c3cc4n(n3)CCC4)=O)CC2)CCS(=O)(=O)CC1 8994,C1(NC(=O)NC(CC(=C)Cl)CO)CCOC2(CCCC2)C1 8995,c1(C(N(C(C)CCNC(c2cnc(Cl)[nH]2)=O)C)=O)ccc(C(F)F)cc1F 8996,c1(N2CCN(C(C(=O)NCC(COC)(C)CO)=O)CC2)ccc(F)cc1OC 8997,CC1(C(F)(F)F)CCCN1C(c1cccc(NCc2ccccn2)c1)=O 8998,C1(NC(CC(n2ccc(C)n2)C)=O)CN(C(C2CC(N3CCCC3)C2)=O)CC1(C)C 8999,C1(CCC)CN(C(c2[nH]c(C)nc2CC)=O)CCN1C(=O)C(C)NC(C)=O 9000,C=CC(C)(CC)C(=O)N(C)CCOCCN(C)C(c1cc(O)cc(F)c1)=O 9001,C(=O)(C(C)C(O)C(C)CC)NC1(C)CN(C(C2(C#C)CCCCC2)=O)C1 9002,c1(CC)ccc(OC)cc1C(=O)NCC1C(CC)CCN1C(c1n[nH]cc1C)=O 9003,C(=O)(CC1OCc2ncccc21)NC(C)CNC(C1C2(CC2)C12CC2)=O 9004,C1(NC(C2CC2Br)=O)(CO)CCCN(C(c2ccc(Cl)cc2)=O)C1 9005,Cc1ccc(S(=O)(=O)NC2CCS(=O)(=O)C23CNC3)cc1Cl 9006,C1(C)(NC(CC2N(C(C)C)CCC2)=O)CCCN(C(C2CCN(C)CC2)=O)C1 9007,c1(-c2c(C)noc2)nc(-c2ccccn2)nn1Cc1ccc(Cl)cc1 9008,C1(C(N2CC(CNC(CCOCC#C)=O)C2)=O)COC2(CO)CC1C2 9009,Cn1nccc1C=CC(=O)NCC1CCC(C(N2CC(O)C(O)C2)=O)CC1 9010,C1(C(=O)OCC)(NC(C2CC(NC(=O)CC3CSC3)C2)=O)CCOC1 9011,CC(=O)CCCC(C)C(=O)N1CCC(C(N2CC3C(C(N)=O)C3C2)=O)C(C)C1 9012,C1(CC(N2CCN(C)C(c3ccccc3)C2)=O)CCN(C(C)(C)C)C2(CC2)C1 9013,C1(CCC)CN(C(=O)CN(C)C(C)=O)CCN1C(=O)C(C1CC1)OC 9014,CCC(CC(=O)NC(CNC(c1nc(C)sc1Br)=O)CCOC)C1CC1 9015,C(=O)(CCS(=O)(=O)C1CCCC1)NCCCN(C(C1CC(OC(F)F)C1)=O)CC 9016,C1(CNC(CSCC)=O)CCN(C(=O)CCn2cc(Br)c(C)n2)C12CC2 9017,Cc1nc2ncccc2cc1C(=O)NCCCCN(C)C(c1nsnc1O)=O 9018,c1(OC)ccc2[nH]c(C(N3CCC(CCNC(C4C=CCCC4)=O)C3)=O)cc2c1 9019,Cc1coc(C(=O)NC2C=CC(CC(=O)NCC3(O)CCOC3)C2)c1 9020,C=C(C)C(O)CC(=O)N1CC=C(CNC(=O)C(CO)NC(N)=O)CC1 9021,c1(C(N(C)CC2(N(C)C)CC2)=O)c(Cl)nn(C)c1Cl 9022,C1(NC(c2ccc(OC)cc2Br)=O)CC2CCCC(C1)N2C(=O)C(C)O 9023,c1(C(N2CC(C)C(NC(c3cccc(Cl)c3)=O)C2)=O)ccc2c(c1)CCCCS2 9024,C#CCCC(C(=O)N1CCC(C)(C(C)C)C1)NC(c1cnc(S)nc1)=O 9025,C1(C(N2C(CNC(c3c(C)cccc3Cl)=O)CCC2)=O)CC2CCCN2C(=O)N1 9026,N1(C(CCNC(CC(C)C)=O)=O)CCC2CCC(NC(=O)CC(C)C3CC3)C12 9027,c1(C(=O)NC2(CC=C)CCN(C(CCOCC#C)=O)C2)ccnc2[nH]c(O)nc12 9028,C1(CC(=O)NCCC2CN(C(CC(C)c3cnn(C)c3)=O)C2)NC(=O)CNC1=O 9029,C(C)(CN=C(NC1CCCCC1)N1CCC(NC(N)=O)CC1)C1C(C)CCCC1 9030,c1(C(N2CC(CNC(CCN(C(C)=O)C)=O)C2)=O)cnc2cc(Br)ccn12 9031,c1(C(N2CC(N(C(c3ccc(C(C)=O)nn3)=O)C)C2)=O)oc(S(N)(=O)=O)cc1C 9032,C1(C(=O)NCC(c2nccs2)C)CCN(C(=O)CN2C(=O)CCC2=O)O1 9033,CC1=Nc2ccccc2C12CCN(C(C1CC3(CC3)CN1C)=O)CC2 9034,c1(OC(C)C)ccc(Cl)c(C(=O)NC(CNC(C2(O)CCSC2)=O)C2CC2)n1 9035,c1(C(N(C(CNC(C2CC(O)(CC#C)C2)=O)C)CC)=O)nc(C)ccc1F 9036,C1(C(=O)NC(C(=O)NC(CN(C(C)C)C)C)Cn2cncn2)CCCSC1C 9037,c1(C(=O)NC2CC(C(=O)NCCCCC#C)C2)ccc(OCCC)c(OC)c1 9038,C(CC[Si](C)(C)C)N(CC(=O)NCCNC(=O)C(CC)OC1CCCC1)CCC 9039,C1(NC(c2cc(C(=O)OC)nn2C)=O)CN(C(c2ncncc2F)=O)CC12CC2 9040,N1(C(C2(C)C(C)(C)C2)=O)CC(NC(=O)CNC(=O)CC2CCCCC2)C(F)C1 9041,c1(C(N2CCC(C3N(C(COC)=O)CC3(C)C)CC2)=O)cc(F)cnc1O 9042,c1(C(C)OCC)nc(C)c(C(=O)NCC(C2CC2)NC(=O)CCCC2(C)N=N2)s1 9043,Cc1ccc(NC(=O)C(F)CC2CN(C(c3cocn3)=O)C2)cn1 9044,C12(C(=O)NCC(C#C)CC3(NC(C)=O)CC3)CC(CN(C(=O)OC(C)(C)C)C1)C2 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9116,CC(C)(CC(F)F)C(=O)N1CCN(C(N2CCN(C(=O)C(C)(C)C)CC2)=O)CC1 9117,O=C1CCN(Cc2nnnn2C2CCCC2)C(=O)N1CCCc1c(F)cncc1F 9118,C1(NC(c2cc(C)[nH]n2)=O)C2CC3CN(C(c4ccnnc4)=O)C1C3C2 9119,C(CC(C(=O)N(C)Cc1nc(C)no1)NC(=O)C=CC1CCOC1)OCC 9120,c1(C(C)C(=O)NC2CC2NC(C2COC2)=O)ccc(C(F)(F)F)cc1 9121,C(=O)(CC(C)Cc1cccc(OC)c1)NCC(CC)(C)O 9122,n1(CC(=O)NCCNC(c2c(CC)c(C)ccc2)=O)nnc2ccccc2c1=O 9123,C1(NC(C)=O)CCN(C(=O)CN(c2ccccn2)CCOCCOC)CC1 9124,C1(C(N(CCC(=O)N(C2CC(OC)C2)C)CC=C)=O)CCC2(CC2)C1 9125,c1(C(=O)NC(CSCC)C(=O)NC(CO)CCO)csc(O)n1 9126,Cc1c(C(=O)NCCCN(CCO)C(C2COCCN2C)=O)c[nH]c1C#N 9127,C(=O)(CC(O)CC(C)C)NC1(CC(=O)NC2CC(CC)C2)CC1 9128,C1(CNC(c2ccc(OC(C)C)cn2)=O)C(C)CCCN1C(=O)C=C(C)C(F)F 9129,C1(C#N)(C(N2CC(C)C(NC(C3(C4CCCO4)CCC3)=O)C2)=O)CC2C=CC1C2 9130,C1(C(=O)NC(C2CN(C(=O)C(C)Cn3ccnc3)C2)C)CC2(C1)CC21CCC1 9131,C(=O)(CCCCN=[N+]=[N-])NC(C(=O)NCC(C#C)CC)COC(C)C 9132,N1(CC)CCCC(ONC(=O)CCC2CC(NC(=O)C(C)=C(C)C)C2)C1 9133,c1(C(=O)NC2CCCC(NC(CCCOC(C)C)=O)C2)ccnc(S(N)(=O)=O)c1 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9170,c1(C(=O)NCC2CC(OC)CN2C(=O)C=Cc2ccncc2)ccnn(C)c1=O 9171,C1(C(=O)NC(CN(CC)CC)C)CCCN(C(=O)N(c2ccsc2Cl)C)C1 9172,N1(C(C(C(C)C)NC(c2cc(OC)no2)=O)=O)CC(O)CC(O)C1 9173,N1(C(c2n[nH]c(C(C)C)c2Br)=O)CCN(C(=O)CC(C)F)C(C)C1 9174,c1(C(=O)NC(CC(C)NC(Cc2c(C)cc(F)cc2)=O)C)cc2n(n1)CCCO2 9175,C1(CCNC(=O)Cc2cc[nH]n2)CC(F)(F)CN1C(c1cc(Cl)c(Cl)s1)=O 9176,C12(NC(c3c(C)occ3)=O)CCCC1N(C(c1ccc(C3CCC3)cc1)=O)CC2 9177,C(=O)(CN=c1[nH]c(N(C)Cc2sccc2Br)nc2c(F)cccc12)NCC(C)C 9178,C12(CNC(C3CC34CCCC4)=O)CCC(CC1)CN2C(=O)COCC1CCCO1 9179,c1(C(C)=O)ccc(C(N2CCN(C(=O)CCCF)C(C)C2)=O)cc1C 9180,C#CCC(CC#C)C(=O)NCC(F)CNC(C1(O)CCCCC1)=O 9181,c1(NC(c2nnnn2C2CCC2)(C2CCCOC2)C)ccccc1SCC(N)=O 9182,Cn1cnnc1CC(=O)N(C1CCN(C(=O)COc2cccnc2)C1)CC1CC1 9183,c1(C(N(CC(C)(C)NC(c2c(C)ccnn2)=O)C)=O)[nH]c2cc(F)ccc2c1C 9184,c1(C(=O)NCC2C(C(=O)NCc3c(OC)cccc3)CCC2)ccc(C)cc1O 9185,C1(OC)(CNC(N2CCCC2C(F)(F)F)=O)CCCCC1 9186,N1(C(C(CC)OC)=O)CCC(O)(C(C)NC(=O)CN2CCC(O)CC2)CC1 9187,c1(C(=O)NC(CN(C(=O)CC2COCCO2)CC)C)cnc(OC)c(Br)c1 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9276,Cc1ccc(CS(N2CC(NC(c3occc3Br)=O)C(F)C2)(=O)=O)cc1 9277,C1(C)(C(=O)OC)CC(C(=O)OC)CN1C(c1cc(Br)ncc1Cl)=O 9278,CS(=O)(=O)c1ccc(O)c(C(=O)NC2(CNC(C3CCC4CC4CC3)=O)CC2)c1 9279,CCC(CC)C(=O)N(CCNC(=O)CCCc1cc(C)sc1C)CCOC 9280,C1(c2n(CCC)nnn2)(NCC2CCCC(C)C2)CCC2(CC1)CSC2 9281,C=CCCCC(=O)NCC(C)CN(C(=O)C=C1CCC(C)CC1)C 9282,c1(C(N2CCC(NC(CCCC(=C)C)=O)CC2C)=O)cnc2[nH]nnc2c1 9283,c1(OCC(=O)NC(CC)(C)CNC(=O)CN2CCCC2C)cc(F)ccc1F 9284,c1(C(=O)NC(CN(C(=O)CC2C(=O)N(C)N=C2C)CC)C)cccc2c1COC2 9285,C1(F)(CNC(c2cnn(CCN(C)C)c2)=O)CC(CNC(C2CC23CC3)=O)C1 9286,N1(C(C2(OC)CCCCC2)=O)CCCC(O)(CNC(=O)CCn2ccnn2)CC1 9287,c1(C(N2CCC(C3(NC(C4CCCSC4)=O)CC3)C2)=O)[nH]c2ccccc2c1Cl 9288,N1(C(C2CC(c3cccc(O)c3)C2)=O)CCC2(CC1)CN(C(c1ccns1)=O)C2 9289,c1(OCC)ccc(S(=O)(=O)NC2CCNCCC2c2ccccc2)cc1F 9290,C1(C)(C(=O)NCC#CCNC(c2n(CC)ccc2)=O)CCCC1O 9291,c1(C(=O)NCC(N(C(C(C)S(N)(=O)=O)=O)C)C2CC2)c(Cl)ccc2ncccc12 9292,C1(c2ccccc2)CCCCC1.c1nc(Sc2ncc[nH]2)no1 9293,c1(CNC(CC(CC)C2CC2)=O)ccc(CNC(=O)CC2CCCC2C)c(F)c1 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9742,c1(C(=O)C(C2CC3C=CC2O3)=O)cnn(C)c1C.C=CCC(CC)O 9743,N1(C(CC(C)(F)F)=O)CCC(NC(=O)CCn2cc(Br)ccc2=O)C(F)C1 9744,CC(CCC(C)(C)C)C(=O)N1CCOCC1CCNC(=O)C(N1CCCCC1)C 9745,N1(C(CN2CCCC(CC)C2)=O)CCC(C(=O)N2CC=CCO2)C1(C)C 9746,N1(C(c2sc(C)c(Br)c2)=O)C2CCC1(CNC(=O)C(C)CS(C)=O)CC2 9747,C1(C)(NC(c2ccnc(C)n2)=O)CCCN(C(c2c(C3CCC3)cnn2C)=O)C1 9748,Cc1ccc(I)cc1C(=O)Nc1ccc(CNC(c2cccc(Br)c2O)=O)cn1 9749,c1(C(N2CCCC(N(C(c3c(C)coc3)=O)CCF)C2)=O)cc(Cl)c(N)cc1F 9750,N1(C(c2nc(CC)sc2)=O)CC2CCC1CN2C(=O)CC1CCCC(C)C1 9751,n1(CC)cc(CC(=O)NC(C)C(N2CCCC2CN(C)C)=O)cn1 9752,N1(C(c2ccc(CC)o2)=O)CCC(O)(C(C)NC(c2cc(C(C)(F)F)n[nH]2)=O)C1 9753,c1(C(=O)NC2C3(CC(NC(C4(CC)CCC4)=O)C3)C2)ccnc(O)c1Br 9754,N1(C(c2coc(C3CC3)n2)=O)CCC(C(N2CCC(n3ccnc3)C2)=O)C12CC2 9755,C=C(C)C(CC(=O)NC1(C)CCN(C(c2cc(Br)c(C)cn2)=O)C1)OCC 9756,c1(CNC(c2cc(CO)[nH]n2)=O)nc2c(s1)CN(C(C1CCCCC1F)=O)CC2 9757,Cc1cnc(S(C)(=O)=O)nc1N(C1CC2CC1CN2)C(=O)CC1CCC1 9758,S(=O)(=O)(c1ccc(Cl)c(C(=O)NC(C)CNC(c2ccc[nH]2)=O)c1)NCCOC 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9777,C1(NC(C(CC)n2ccnc2)=O)CC2CC1CN(C(c1cc(Cl)sc1Cl)=O)C2 9778,c1(SC)ccc(Cl)c(C(N2CC(NC(=O)CCc3cccs3)CCC2C)=O)c1 9779,c1(C(N2CCOCC(NC(C3C(C)CC(=O)N3)=O)C2)=O)cc2n(n1)CCCN2 9780,CC1CN(C(C2(CO)CCOC2)=O)CC1CC(=O)NCC1=CCCC1 9781,C1(CCOC)COCCC1Nc1cncc(CO)c1 9782,N1(C(c2cn(CCC)nc2)=O)CCCC(C(=O)NC2CN(C)CC23CC3)(CC)C1 9783,C1(NC(C(=C)CN(C)C)=O)(CN(C)C)CCCCC1C 9784,C12(CO)CCCN(C1)C(=O)C1C(C)(C1)C(=O)N2.c1(C(=O)OCC)ccc(F)cc1 9785,C1(C(N(CC(N2CC(c3ccon3)C2)=O)CCOC)=O)CC2CCC(C1)O2 9786,C1(NC(C(C)(C)OC)=O)CCCCCC1NC(c1ccnn1-c1ccncc1)=O 9787,C(=O)(C(CCC1CCCO1)N(c1nc(Cl)cs1)C)NCCCSC 9788,c1(CC(C(=O)NC(c2ccccc2)Cn2ccnc2)O)ccccc1Br 9789,C=CC(CCC)CC(=O)NC1CCC(O)CN(C(c2nccn3ccnc23)=O)C1 9790,c1(C(=O)NCCN(C(c2cnc(Cl)[nH]2)=O)C2CC2)c(C(F)F)nc2n1CCCC2 9791,C(=O)(NNc1cc([N+](=O)[O-])ccc1Br)n1c(-c2n(C(C)C)cnc2)ncc1 9792,C1(CNC(=O)COCC2CC2)(CNC(C2CC3C=CC2C3)=O)CC12CCC2 9793,C(C(C(C)C)NC(c1cc(CNC(=O)Cc2coc(C)n2)[nH]n1)=O)OC 9794,CC1=NNC(=O)C1CC(=O)NCC12CC(NC(c3cc(C4CCC4)on3)=O)(C1)C2 9795,c1(CN2CCC(N(C)C(c3ccoc3)=O)CC2)cccc(Cl)c1C#N 9796,c1(OC)ccc2nc(C(=O)NC3(C)CCN(C(=O)Cc4csnn4)CC3)cn2n1 9797,Cc1sc(C)c(C(=O)NC2CN(C(C3CC(=O)N(C4CC4)C3)=O)CC2C)c1C#N 9798,C=CC(C)(CC)C(=O)NC1C2CN(C(=O)CCOc3ccccc3C)CC12 9799,C1(NC(C2CC(Sc3ccncc3)C2)=O)CCOCC1CNC(c1cccs1)=O 9800,C1(CNC(c2n(C=C)ncc2)=O)CN(C(C2(C)CC(F)C2)=O)CCN1C 9801,Cc1cc(C)c(C(=O)NCC2(O)CCN(C(C3CCCN(C)C3)=O)C2)c(=O)o1 9802,N1(C(=O)OC(C)(C)C)CCCOC(CCOC(C2CC(O)C(F)C2)=O)C1 9803,C1(C#N)(C(N2CCC(N(C(=O)Cn3ccnn3)CCC)CC2)=O)CCCOC1 9804,O=C(C1CCc2c[nH]nc21)NC1CN(C(c2cnco2)=O)C2(CCCC2)C1 9805,C(c1ccsc1)=CC(=O)NC1(C(=O)NC2C=CCC2)C(C)C1 9806,CC(C)(C(=O)NC1CCCC1NC(=O)CC1COCC1O)NS(C)(=O)=O 9807,Cc1nccn2ncc(C(=O)NC3(CNC(C45CCCN4CC(O)C5)=O)CC3)c12 9808,N1(C(=O)OCC)CCCC(C(=O)N(CCCNC(c2cc(C#N)cs2)=O)C)C1 9809,C12(COC)CC(NC(=O)C=Cc3ccc(C)s3)(CN1C(c1cnc(C)nc1)=O)C2 9810,c1(C(=O)NC(C(CO)NC(C(COCC)C)=O)C)cccc2nc(O)n(C)c12 9811,c1(OC)cn(C)c(C(N2CCC(C(F)CNC(C3CC3C)=O)CC2)=O)cc1=O 9812,c1(OC)cc(COc2c(Cl)nc(Cl)n2C)ccc1C 9813,c1(CC(=O)CCl)ccccc1C1CC1C(=O)Oc1ccsn1 9814,CC1CN(C(=O)CC2CCCN2C(C2CC(=O)OC2(C)C)=O)C(C)C1C 9815,C1(CNC(CN(C)CC2CCCC2)=O)CCN(C(C2CCSC2)=O)CC1(F)F 9816,N1(C(CN(C)C)=O)CCC2CC2(C(=O)N(C)C2CC2)CC1 9817,c1(SCC(=O)NC2C3CN(C(C(CC)(C)OC)=O)C2C3)nc2ccccc2s1 9818,c1(C(=O)NC(C(=O)NC(CNC(=O)OC)C)C)ccc(C)cc1 9819,NC(=O)CC(O)C(=O)N1CCCC(NC(=O)COc2ccc(Cl)nc2)CC1 9820,N1(C(COCCCOC)=O)CCCN(C(=O)CSCc2cccs2)C(C)C1 9821,n1(CC)c(CN2CCC3(CN(C(=O)C(F)F)C3)C2)nc2ccccc12 9822,C1(C(=O)NC(=O)C(CC2CC2)CN(C2CC2)CC)CCC(C(=O)OC(C)(C)C)CC1 9823,N(C(=NCCCCl)NC(c1nc2c(s1)CCC2)C)CC1(OC)CC1 9824,C(=O)(C1=NOC(C)C1)NCC(Cc1ccccc1)NC(C1OCCN(CC)C1)=O 9825,C1(C(=O)NC(c2cnn[nH]2)C)CN(C(C2(O)CC(CF)C2)=O)CC1C 9826,c1(C(=O)NCCCC(=O)OC)cnn2c(C(F)F)cc(C)nc12 9827,CC1=C(C(=O)NC2(C)CN(C(=O)CC3=CCOCC3)C2)COCC1 9828,c1(N2CCC(C(C)(C)C)C2)nnc(CS(N)(=O)=O)n1Cc1nc(C2CC2)cs1 9829,CC1CC(CNC(c2cncn2C)=O)CCN1C(=O)Cc1cc(Br)cs1 9830,C1(O)(CC(N2C(CCCC)CCC2)=O)CCN(C(c2ccc(F)nc2C)=O)CC1 9831,c1(OC)ccc(C(CNC(=O)CC2CC23CC3)NC(=O)C(C)N(C)C)cc1 9832,c1(NCCC2CCC(C)O2)ccc(S(=O)(=O)NCc2c(F)cccc2F)cc1Br 9833,C1(C(=O)NCC(C(C)C)NC(C2C(=C)C2)=O)CCN(C2CCSC2)CC1 9834,C=C(Cl)CC(C(=O)NCC1(CC2CC2)CC1)NC(C1C=CC1C(=O)OC)=O 9835,N1(CC(n2cc(CCCC#N)nn2)C)CCC(=C(F)F)CC1 9836,N1(C(C2CN(C(C)=O)C2)=O)CC2CCCC(NC(C3(C)CCC(C)C3)=O)C2C1 9837,N1(C(C(c2ccccc2)C)=O)CCCC(NC(=O)C(F)(F)C2(O)CCC2)CC1 9838,c1(C(N(C2CCCN(C(=O)Cc3cc[nH]c(=N)c3)C2)CC)=O)ccc(C)c(Cl)c1 9839,C(=O)(C(C)C(C)NC(=O)CSc1nc[nH]n1)NCc1c(C(C)C)ocn1 9840,C(=O)(C#CC1CCCOC1)N1C(C)CC(NC(c2c(C)ncn2C)=O)C1 9841,C1(C)(CC)C=C(C(=O)N2CCC(CC)(NC(c3snc(C)c3N)=O)CC2)C1 9842,c1(C(=O)NCCCCNC(c2coc(O)n2)=O)ccc2occc2c1 9843,N1(C(COCC=C)=O)CCN(C(=O)COCC(C)(C)C)CC1CCOC 9844,c1(C(=O)NC23CC(NC(CCc4cc(C)[nH]n4)=O)(C2)C3)ccc2c(n1)CCCC2 9845,CC1CC(NC(c2cnc(Cl)[nH]2)=O)CN1C(=O)CCNC(c1ccco1)=O 9846,C1(NC(c2n(CC)ncn2)=O)CCC2(CC1)CC2NC(c1cc([N+](=O)[O-])c[nH]1)=O 9847,C1(C(=O)NC(CC)(CC)CCNC(c2cccs2)=O)CCc2nn(C)cc2C1 9848,C1(NC(N)=O)C2CCC(NC(=O)OCC(=O)NCc3cccs3)C1CC2 9849,c1(C(=O)NC2CC(CNC(C(C)SC)=O)C2)ccc(OCC2CCC2)cc1 9850,CCCCS(=O)(=O)N1CCCC1C(N1CCCC1CNC)=O 9851,C12(OC)CCC(C(N3CCC(C)(CNC(C4C(C)(C)C4(F)F)=O)C3)=O)(CC1)C2 9852,C1(C(=O)NC(CC)(C)CC)CN(C(=O)C(C)Nc2ccccn2)CCC1O 9853,c1(C(=O)NC2(CO)CCN(C(C3C(C)C3)=O)C2)ccc(Cl)c(F)c1N 9854,c1(NCC2(CCCC)CC2)ncc(C)cc1S(=O)(=O)NC(c1cccc(Br)c1)C 9855,C(=O)(C(CCC(C)C)NC(=O)Cc1cc[nH]c1)N1CCC(C)(OC)C1 9856,C1(CNC(CCc2ccc(C)nc2)=O)CN(C(=O)Cc2nc[nH]n2)CC(C)(C)O1 9857,c1(C(N2CCC(NC(c3ccc(C(N)=O)cc3)=O)C2)=O)ccc(O)c(F)c1 9858,C1(CC=C)(C(=O)NCCc2ncc(C)o2)CCN(C(c2cc(Cl)cn2C)=O)C1 9859,C1(NC(C(C)O)=O)CN(C(c2cccc3ccccc23)=O)C2(CCCC2)C1 9860,C#CC1CC2(C1)NC(=O)N(c1ccc(OCC)c(Cl)c1)C2=O 9861,N1(C(CC(=C=C)C)=O)CCN(C)C(CNC(=O)C=CC(N2CCOCC2)=O)C1 9862,C(C)(CCC(=O)NC1CN(C(c2ccncc2C(F)(F)F)=O)C1)OC 9863,Cc1nc(N)cc(SCCOC2CCC2)n1 9864,C1(C(N(C)CC2N(C(CCC(C)C#N)=O)CCC2)=O)CCS(=O)(=O)C12CCC2 9865,CCN=C(NCC12CC(C)(CO1)C2)N1CCCC2(CCSC2)C1 9866,C12(NC(c3c[nH]c(C(F)F)c3)=O)CC(C1)N(C(c1cnc[nH]1)=O)C2 9867,C1(Nc2cc(OC)ncn2)CN(C(C23CC(C2)C3)=O)CC12CC2 9868,c1(OCC(=O)NCC(C2(O)CN(C(=O)C(O)C3CC3)C2)(C)C)ccccc1C#N 9869,c1(C(=O)NCC(CNC(c2nnn(C)n2)=O)(C)C)cnn2cc(Br)cnc12 9870,CC(CC(F)(F)F)C(=O)NCC(CO)NC(c1cnc2sccn12)=O 9871,N1(C(C2C(C)=CCS2)=O)CC2CC(C1)C(CO)C2NC(C1CCC(C)=C(C)C1)=O 9872,CCCCC(C)C(=O)N1CC(C(N)=O)(CNC(C2CCC=CO2)=O)C1 9873,c1(C(N2CCN(C(C3(CC)CC3)=O)CC2CO)=O)cccc2c1CCS2(=O)=O 9874,CC1CC(CC(=O)NCC2C3CN(C(C4CS(=O)(=O)C4)=O)CC23)CCC1C 9875,Cc1ccc(CC(N2CCC(F)(CNC(C3(C)CC3(F)F)=O)C2)=O)cc1Br 9876,C1(NC(=O)CC2CC3CCC2C3)CCN(C(=O)CC2(CO)CCC2)CCC1CO 9877,c1(C(=O)OC(C2CCN(C(=O)CC3C4CN(CC)CC34)C2)=O)cc(F)cc(Cl)c1 9878,N1(C(C2N(C)CC(O)C2)=O)CCC2(CCN(C(=O)C=Cc3nccs3)C2)C1 9879,N1(C(COCc2c(C)cccc2)=O)CCN(C(=O)Cc2ncoc2C)CC(O)C1 9880,N1(C(C(C2CCOC2)NC(C2C(CC(C)C)C2)=O)=O)CCC2(C=CCO2)CC1 9881,Cc1cnccc1C(C)CNC(=O)C(=O)NC(C12CC(CO1)C2)C 9882,C(CN=C(NC1CCC1)N(C)CC1CCCN1C)c1ccc(OC)cc1 9883,n1(CC)nc(C)c(CC(=O)Nc2ccc(OCCOCCO)cc2)c1C 9884,N1(C(CCCOCC)=O)CCCC(C)(C)C1CNC(C1CC=CC(O)C1)=O 9885,c1(C(N(CC(=O)NC(CNC(C=CCOCCOC)=O)C)C)=O)ccccc1 9886,CC1C(C(=O)NC(C(=O)NCC(C)(C)CN=[N+]=[N-])C2CCOC2)=NOC1C 9887,Cc1cc(C(N2CCCC(C3CCCCN3C(=O)C#CC(C)C)C2)=O)[nH]c1C 9888,N1(C(C2CC=CC(NC(CCOCCOC)=O)C2)=O)CC2CC(C1)N(C)C2 9889,C(=O)(CC1OCc2ccccc21)NCC1CC(NC(c2c(CC)csc2)=O)C1 9890,C12(C(N3CCC(F)(C(=O)NCC4N(C)CCCC4)C3)=O)CCCC1C2(F)F 9891,C1(NC(=O)CCc2ccncn2)C2CC3CN(C(=O)C4=COCCC4)C1C3C2 9892,Cc1ccccc1CNC(=NCC1CCSC(C)C1)NC1CC1 9893,c1(NC)snc(C)c1C(N1CC(CNC(=O)C=CSC)C1)=O 9894,C1(c2cccc(OC)c2)CN(C(=O)C=C2CCC(C)C2)CCN1C(=O)CNC=O 9895,C1(NC(C2(CC=C)CN(C(c3ccncc3)=O)C2)=O)COC2COCC12 9896,C(=O)(CC(C)(C)c1ccccc1)N(CCCNC(C1(CCF)CC1)=O)C 9897,c1(OC)ccc(OCC(N2CCC(C(C)(C)NC(c3cn(C)nn3)=O)C2)=O)cc1 9898,N1(C(CC(C(F)F)NC(c2cc(C(N)=O)[nH]n2)=O)=O)C(CO)CC2CCCC12 9899,Cc1ccncc1C(C)(C)C(=O)NC1CCC(NC(C2CCCOC2)=O)CC1 9900,c1(C(=O)NC2C(C(N(CC)Cc3cccc(Cl)c3)=O)C2)ccc(Cl)c([N+](=O)[O-])c1 9901,N1(C(CC(C)C)=O)CCCC2C1CCCN2C(=O)Cc1ccn(C2CCCC2)n1 9902,c1(N2CCC(C3(OC(CC(CCC)C)=O)CC3)C2)cc(OC)c([N+](=O)[O-])cc1Cl 9903,c1(C(C(=O)NCCC(CCNC(C2(OC)CCCC2)=O)C)=O)cc(F)cc(Cl)c1 9904,C1(NC(CCNC(N)=O)=O)CN(C(=O)CSC2CCCCO2)CC(F)(F)C1 9905,C1(F)(CNC(C(C)=C2CC2)=O)COCCN(C(C2(c3ccc(F)cc3)CC2)=O)C1 9906,c1(OC)ccc(C(CNCc2cc(C(C)C)n(C)n2)N(C)C)cc1 9907,N1(C(c2cccc3ccn(C)c32)=O)CCOC2(CCN(C(C3CC3(F)Cl)=O)C2)C1 9908,N1(C(C)=O)CCOC(C(N2CCC(NC(=O)Cc3ncc(C)o3)C2C)=O)C1 9909,CC1(C)CCCCC1(C)NC(=O)CNC(C1CCC(C#N)CC1)=O 9910,CCC(CNC(=O)CCCCCn1cc(C(C)(O)CSC)nn1)CC(F)F 9911,Cc1noc(C)c1C(=O)NCC12CC1CN(C(=O)Cc1cccc(C(F)(F)F)n1)C2 9912,C=CC1(C(=O)Nc2ccc(OC)cc2)CCN(C(C2CC3(C2)CC(C)C3)=O)C1 9913,c1(SC)ccc(C(N2CC(NC(c3ncn(C)c3C)=O)C(C(F)F)C2)=O)c(Cl)c1 9914,N1(C(C(C)CF)=O)CCC2(CCCCC2NC(c2cc(F)cc(Cl)c2)=O)CC1 9915,Cc1nn[nH]c1Cn1cc(COC2CCOCC2)nn1.C12CCN1C(=O)CO2 9916,N1(C(C(CC)OCC)=O)CC2CCC(C1)C(NC(c1c(C)nn(C)c1Cl)=O)C2 9917,C1(CO)CCC(CNC(c2nnnn2CCCF)CC2CCOC2)CC1 9918,CC1CCCCC1(CNC(=O)CCC(=O)c1ccccn1)NC(c1cnsc1)=O 9919,c1(C(N2C(CCNC(C(C(C)O)N(C)C)=O)CCC2)=O)ccc(Cl)c(N)c1 9920,c1(C(=O)NCC2CCC2NC(C2C(F)(F)C23CC3)=O)cc(C(F)(F)F)ccc1F 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9939,CN=c1[nH]cc(C(=O)NC2C=CC(C(=O)NCC(CO)OC)C2)o1 9940,C1(NC(=O)Cc2cn[nH]c2)CC12CCN(C(c1ccc(O)cc1Cl)=O)CC2 9941,N1(CC)CCN(C(=O)C=CC(C)NC(=O)C(F)C(C)(F)F)CC1C 9942,CC1=C(C(=O)NC2COCCC2NC(=O)C=Cc2cnc[nH]2)CCC1 9943,C(=O)(CCCCCC(=O)N1CC(NC(=O)C(F)=C2CCC2)C(C2CC2)C1)OCC 9944,c1(C(=O)NCCC2CCC(NC(C3(COC)COC3)=O)C2)c(C)ccc(Cl)c1O 9945,N1(C(c2cc(C)nn2CC(F)F)=O)CCC(F)C(NC(C2CCCC2)=O)C1 9946,Cc1c(C(N2CC(CCNC(=O)C(C)(C)C)OC(C)C2)=O)[nH]c2c1C(=O)CCC2 9947,N1(C(c2ccc(CC)c(CC)c2)=O)CC2CCN(C(c3cccn3CC)=O)C2C1 9948,C1(CNC(=O)C=C2CC2)CC(F)CN1C(=O)CCC1CCCO1 9949,N1(C(C=C(C)Cl)=O)CCN(C(c2cccn(C)c2=O)=O)C(C(C)(C)C)C1 9950,CCCCC(C(=O)N1CCC(N(C)C(C23CC(CC)(CO2)C3)=O)CC1)NC(N)=O 9951,C1(C(N(C(CNC(CN(C)C2CC2)=O)C2CC2)C)=O)CC2CC1CO2 9952,c1(C(N2C(C)(CNC(=O)CC3(O)CCCOC3)CCC2)=O)cccc(N=[N+]=[N-])c1 9953,Cc1[nH]nc(C(F)(F)COC(=O)CSC=Cc2ccoc2)c1C(=O)OC(C)(C)C 9954,C(=O)(CC(C)C(F)F)NC(CC)(C)CCNC(=O)Cc1n[nH]c(C)n1 9955,N1(C(c2cc(C)c(F)cc2)=O)CC2CC1CCN2C(=O)Cn1cncc1C 9956,S(=O)(=O)(c1ccc(Br)c(OC)c1)Nc1cc(OC)c(Cl)c(NC(c2cccs2)=O)c1 9957,C1(NC(C2CC3CCC(C2)C3O)=O)CC2CN(C(C3CC(O)C3)=O)CC2C1 9958,CC1CCC(C(N2CC(CO)CC2CO)=O)CN1C(=O)Cc1cc[nH]c1 9959,N1(C(c2cc(C(C)C)no2)=O)CCC(C(N2CCCCC(C)CC2)=O)CC1(C)C 9960,N1(C(=O)C=C(Cl)Cl)CCC(C2CCN(C(C3CC3[N+](=O)[O-])=O)CC2)C1 9961,C1(C(=O)NC2(C)CCC(C)C2)CC2(CC(NC(C3(O)CC4CCC3C4)=O)C2)C1 9962,c1(C(=O)NCC2(F)CC(NC(CC3CC(=O)NC3)=O)C2)csc2nnsc12 9963,C1(NC(C2C(=C)CC2)=O)CCC2CC1CN2C(c1c[nH]ccc1=O)=O 9964,C1(C(=O)NC(C(=O)OC)C)CCC(C)(C)N(C(=O)Cn2cccnc2=O)C1 9965,C1(CC)CN(C(=O)Cc2cccc(C)c2Cl)CCC1NC(c1ncc(C)cn1)=O 9966,N1(CC(=O)NCCOCC)C2CCC1CN(C(c1ccccc1OC)=O)CC2 9967,C12(CNC(=O)CC3CC3)CCCC1N(C(=O)CN1CCCCC1)CCC2 9968,C=C1Cn2c(C(=O)NCC3(C)CCN(C(=O)C(=Cc4c[nH]cn4)F)C3)nnc2S1 9969,CCC(C)CC(C(=O)Nc1ccc(OC)cc1C)NC(=O)CC1(O)CCOCC1 9970,C(C)(C(C)(C)CO)NC(C1C(CNC(C2(CC)CCCC2)=O)CCC1)=O 9971,Cc1nn(CC(N2CCC(NC(=O)COCC3CCOC3)C2C)=O)cc1[N+](=O)[O-] 9972,C1(NC(c2cnsc2)=O)CC2CCC1N2C(=O)COc1ccc(Cl)nc1 9973,c1(C(=O)NC(c2cncnc2)C)cccc(CNC(C2CCC3(CC3)C2)=O)n1 9974,C(=O)(C1=CCC(C)(C)CC1)NC1CC(CNC(c2c(C)[nH]nc2C(F)F)=O)C1 9975,N1(C(CCCOCCC)=O)CC(C)CCC1CNC(=O)CNS(=O)(=O)CC 9976,N1(C(C(C)C#N)=O)CC(F)(F)CC1CCNC(c1ccc(C(C)(C)C)cn1)=O 9977,C(CCCC(=O)NC1CN(C(c2snnc2C2CC2)=O)CC1O)NC(N)=O 9978,N1(C(C2CCN(C(C(n3c(C)ccn3)C)=O)C(C)C2)=O)CC2CCC1C(O)C2O 9979,C=CCN=C(NC1CC12CCC2)N1CCCC(c2ccccc2)C1 9980,Cc1cc(C)n(C(C)CC(=O)NCCC(C)NC(=O)CSCc2ccccc2)n1 9981,C(=O)(CC(=O)NCC1CCC1NC(C1(C2CCCCO2)CC1)=O)NCC 9982,N1(C(c2c(CC)oc(C)c2)=O)CCCC(NC(=O)C=C2CCCCC2)C1CC 9983,C(=O)(C1=CC2(CCOC2)C1)NC(CCC(=O)NCc1c(OC)n(C)nc1)(C)C 9984,c1(C(N2CC(NC(CCC=CC)=O)C3(C2)CC3)=O)ccc2sncc2c1 9985,CCC(CC(=O)N(C1CC1)CC1CCCN1C(=O)CCc1nc(C)cs1)SC 9986,C(=O)(C1=CC2CCCCCC12)NCC1(CNC(c2ccc(C)o2)=O)CC1 9987,N1(C(CCCN(C)C)=O)CC(C2CCCN(C(=O)C=CS(C)=O)C2)C1 9988,Cc1cc(C(=O)NCCC(C)NC(=O)C(C)C#N)n[nH]1 9989,N1(C(CN(C2CCCCC2)C)=O)CC(F)(F)CC1(C)CNC(c1csc(Cl)n1)=O 9990,c1(CNC(c2cc(C)ncc2)c2nnnn2-c2ccccc2Cl)cc(Cl)cc(Br)c1 9991,c1(C(N2CC(CNC(C3(CF)CCC3)=O)C3(CC3)C2)=O)cnc2n1CCCC2 9992,C1(NC(c2c(C)nsc2)=O)CN(C(=O)C(C)N(C)Cc2ccccc2)CC1(C)C 9993,CCC(C)(C)C(O)C(=O)N1CCC(NC(=O)Cc2sccc2Br)C1 9994,N1(C(CCOCCOC)=O)CCCC12CCN(C(C1CCCCC1C)=O)CC2 9995,c1(OC)ccc(C=CC(=O)NCC2CN(C(C3OCCC3C(C)C)=O)C2)nc1 9996,C(=O)(CC1CCC(=O)c2ccccc21)N(C(C)CNC(=O)COCC1(F)CC1)C 9997,c1(C(N2CC3(CC(CNC(C4(CC)CC4)=O)OC3)C2)=O)cnc2c(c1)CCCO2 9998,c1(CC(=O)NC(CCN(C(C2N(C(C)=O)CCC2)=O)C)C)cccc(Br)c1 9999,CC(C(=O)N(C1CN(C(c2nn(CC(F)(F)F)cc2Cl)=O)CC1O)C)C(C)(F)F 10000,CCCC(CCC)C(=O)NC1CCC(C)N(CC2(c3cccc(C#N)c3)CC2)C1 10001,C1(C(=O)OC)C(NC(=O)C(=O)NCCSc2nnc(C)o2)C2CC1C(O)C2O 10002,N1(C(C2OCCC(C)(C)C2)=O)CCC2(C=C(C(=O)N3CCC3C3CCOC3)C2)C1 10003,C(CCCC(=O)N1CCC1CNC(C1(F)CCCOC1)=O)N(C)C 10004,c1(CC)c(N2CC(NC(C3CC(=O)N(CC(C)C)C3)=O)CCC2C)ncnc1Cl 10005,c1(C(N2CCN(C(=O)Nc3c[nH]ccc3=O)CC2)=O)ccnn2ccnc12 10006,N1(C(COC2(C#C)COC2)=O)CC(C(N2CCCCCC2)=O)C(C2CC2)C1 10007,c1(N(C)Cc2ccncc2F)cccc(S(=O)(=O)NC2CSC2)n1 10008,C1(C(N2CCC(C)(NC(=O)CCCC(N)=O)CC2)=O)CC(F)(F)C12CCC2 10009,c1(NC(C(C)(C)c2ccsc2)=O)cccc(NC(c2cc(Cl)c[nH]2)=O)c1 10010,C(=O)(CS(=O)(=O)C(C)(C)C)NC1C(C)CN(C(c2scnc2C(C)(C)C)=O)CC1 10011,c1(C(N2CCOCC(NC(c3cccc(SC)c3)=O)C2)=O)ccc2c(c1)CCC2 10012,N1(C(c2cc3nc(C)oc3cc2)=O)CCc2ccccc2C1CNC(=O)C1CC1 10013,C1(NC(c2c(OCC)nccc2)=O)CC(O)CN(C(C23CCCC(CO2)C3)=O)C1 10014,N1(C(C2(CC)COC2)=O)CCCCC1C1(NC(=O)CN2CC(C)(C)C2)CC1 10015,c1(C(=O)NCC2CC(F)(CNC(c3cc(C)oc3C)=O)C2)cc2n(n1)CCOC2 10016,N1(C(C2(COCC)CC2)=O)CCCC1(CNC(=O)CC1COCC1(C)C)COC 10017,C1(C)(C(=O)NCC(CC)NC(c2cccc(C(C)(F)F)n2)=O)CCC(=O)NC1 10018,Cc1cnccc1C(C)C(=O)NCC1CN(C(=O)CC2CCOC(C(C)C)C2)C1 10019,c1(CNC(=O)OC(C)(C)C)ccc(CNC23CC(C2)NC3=O)cc1 10020,C(CCCC(C)NC(C1CCCCC1)c1ccccc1)NC(C(C)CC1CC1)=O 10021,c1(C(C(=O)NCCCN(C(=O)C2=COCC2)C(C)C)C)ccc(C(F)F)cc1 10022,C(=O)(C1=NOC(CNC(c2ncsc2C)=O)C1)NC1CCN(CCC)C1 10023,C(CCSC)(C(=O)NC(c1nccc(C)n1)C)NC(c1cc(OC)ns1)=O 10024,C(=O)(CC(C)(C)C(=O)NC1COCCC1NC(c1cc(CC)c(C)s1)=O)OCC 10025,c1(CCC(=O)NCCC(O)CNC(C2(CO)CCCC2)=O)ccc(Cl)cc1Cl 10026,N1(C(C=CCCC)=O)CCCN(Cc2cn(CCCC(=O)O)nn2)CC1 10027,N1(C(CCC2CCN(C(C3(OC)CCOC3)=O)CC2)=O)CC2C(C1)C2(F)F 10028,C1(CNC(=O)COC(F)(F)F)C2CN(C(c3c[nH]cc3Br)=O)CC12 10029,C1(NC(C(CCF)NC(c2cccc(OC)c2)=O)=O)C2C=CC(C2)C1CO 10030,c1(C(=O)NC2C(CNC(CC(C)c3ccncc3)=O)C2)nnc2n1CCCCC2 10031,n1(CC(=O)NCCOC2CCCCC2)cccnc1=O.C12CCC(C1)NC2=O 10032,CCC(CC1CCCC1)C(=O)NCCNC(=O)CNC(=O)Nc1ccc(Cl)cc1 10033,CS(=O)(=O)C(CNC(=O)C=Cc1ccc(F)cc1)CNC(=O)Cc1ccsc1 10034,n1(CC)nnc(C(=O)N(CC(C)(C)C(=O)NCCc2nnc(C)n2C)C)c1C 10035,C1(C(=O)NCc2c(C(=O)NCC(C3CCC3)OCC)n[nH]c2)CCCCC1C 10036,N1(C(Cc2c(C)ccs2)=O)CCOC(CCC(=O)O)C1.N12CCC(CC1)C2 10037,N1(C(C23CC(CCC)(C2)C3)=O)CCN(C(c2c(C)nn(C)c2Cl)=O)CC1C.C1CC1 10038,C1(C(CNC(C2C(C(=O)OCC)C2)=O)O)(C(=O)OC)CCCC1 10039,N1(C(C2(C)CCC2)=O)CCC2(CCCN2C(=O)CS(=O)C(F)(F)F)C1 10040,c1(CC)nc(CNC(=O)C(=O)N(C(c2ccco2)CO)Cc2ccccc2)cs1 10041,c1(CC)cccc(CC)c1CC(=O)N(C)CC1CCCN1C(C1CCOC1C)=O 10042,N1(C(c2c(CC)nco2)=O)CC2OCCN(C(=O)C(C)C(O)C(C)C)C2C1 10043,CC1(CNC(C2CC(O)C(F)C2)=O)CCN(C(=O)CCn2cnccc2=O)CC1 10044,Cc1cc(NC(c2nccnc2Br)=O)n(C2CCOC2)n1 10045,N1(C(C2(NC(C)=O)CC2)=O)CCCC(N(C(=O)C(C)C)CC(C)C)C1 10046,CC1(CNC(c2ccnc(S)c2)=O)CN(C(c2ccc(CO)c(F)c2)=O)CCO1 10047,C1(C)(CC)C=C(C(=O)NC2CC2NC(C2(C(=O)OC)CC2)=O)C1 10048,C1(C2(NC(c3cc(C(N)=O)no3)=O)CC2)CCCCN1C(=O)CC1C=CCC1 10049,c1(OCC(=O)NC(CNC(c2ccc(NC(C)=O)cc2)=O)C)ccc(F)cc1O 10050,C1(C(=O)NCCNC(=O)OCC)CC=CCN1C(c1ccsc1C)=O 10051,C(=O)(CCCCCCCC1CC1)NC(C)CNC(c1c(Cl)cnn1C)=O 10052,c1(-c2cc(C(N(C(CCNC(CN3C(C)CC3)=O)C)C)=O)on2)cccc(F)c1 10053,C1(C)(CCNC(C(C(C)C)OCC)=O)CCN(C(=O)C(C2CCCCC2)F)CC1 10054,O=C1CCC(C(=O)NC2(CNC(=O)C3=C(Cl)CCCC3)CC2)c2ccccc2N1 10055,N1(C(=O)C(F)(F)C2CC2)CCC2(CC1)CCN(c1nc(O)c3c[nH]nc3n1)C2 10056,C(C1=CCN(CC(=O)NC2CCCCCC2)CC1)NC(C1C(OC)CCCC1)=O 10057,C(=O)(C(C)CC(C)(F)F)NC1C(NC(c2c(C)oc(Br)c2)=O)CCOC1 10058,C1(NC(c2c(CC)onc2C)=O)CCCN(CCOc2ccc(Cl)cc2Cl)CC1 10059,C(CO)(C(C)(C)C)NC(CC1CC(C(=O)Nc2c(OC)ccs2)C1)=O 10060,C(C(C)C(=O)NCC1(C(C)(C)O)CN(C(=O)CCSC2CCCC2)C1)OCC 10061,CCCCC(C)CCC(=O)NCCNC(=O)C(c1ccccc1)n1cccn1 10062,C1(CNC(COCC=C)=O)CCC2CN(C(c3ccncc3CC)=O)CCC2C1 10063,C1(=CC(N2CC(NC(=O)C=C3CCC3)CC(C)C2)=O)CCOc2ccccc21 10064,c1(CC)ccc(C(C)C(=O)NCC(O)CNC(=O)CCc2cncs2)cc1 10065,c1(CC(=O)N(C(CNC(c2c(CC)n[nH]c2)=O)C2CC2)C)cc(C)ccc1Br 10066,c1(CC(=O)NC2CN(C(c3cc[nH]n3)=O)C3CC23)ccc2c[nH]nc2c1 10067,N1(C(c2c(C)cc(CNC(CC3ON=C(CC)C3)=O)o2)=O)C2CCC1CC(F)C2 10068,C#CCCCC(C(=O)NCCSC)N1CCC(COC)C1.n1(C)cccn1 10069,C(CC(F)(F)F)N(C)CCN(C(=O)CCNC(c1noc(-c2cccs2)n1)=O)C 10070,c1(NC(C)=O)cccc2c1CCCN2C(C1OCCC1C(=O)O)=O 10071,C1(NC(C)=O)CCC12CN(C(C1CCC(C(N)=O)CC1)=O)C2 10072,Cc1nc2ccc(C(=O)Nc3cc(Cl)c(OC(F)F)c(Cl)c3)cc2n(C)c1=O 10073,C1(C)(OC)CCCN(C(C2(F)CCN(C(=O)CCCC(=O)OC)CC2)=O)CC1 10074,c1(-n2cc(CCCC)nn2)cccc(C(=O)NCC(=O)N(CCC)CCNC)c1 10075,C(=O)(C(C)(C)NC(=O)C(F)(F)F)NCC(C(C)C)NC(=O)C(C(C)C)C1CCC1 10076,N1(C(c2cc(C)c(O)cc2)=O)CC(F)(F)CC1(C)CNC(C1CCC1(C)C)=O 10077,N1(C(c2nc(C(N)=O)sc2)=O)CC(CNC(C2CS(=O)C2)=O)N2CCC1C2 10078,CC1(C)CC(NC(c2ccc(C(C)(C)C)o2)=O)CC(O)C1 10079,c1(C(=O)NCC2CCC(CNC(C3CC34CCOC4)=O)CC2)ccc(F)c(Cl)c1 10080,c1(C(N2CC3C(NC(C4CCC(C)O4)=O)(C3)C2)=O)cc2c(Cl)cncc2s1 10081,CS(=O)c1ccc(CC(=O)NCC(O)CNC(c2conc2C2CC2)=O)cc1 10082,C1(NC(CCC2CCCN(C(c3c(CC)occ3)=O)C2)=O)CNC(=O)C12CC2 10083,CCCC(O)CC(=O)NC(CN(C)C(c1nc(C)ccc1F)=O)CC 10084,C1(CC=C)(NC(=O)CC2CCCN2C)CCN(C(=O)CN(C)C(C)=O)C1 10085,c1(C(=O)NC2CC3(C(N4CC(N5CCC5)C4)=O)COC2C3)cn2ccccc2n1 10086,CC(CCC(C)(C)C)C(=O)N1CC(C2CC2C(=O)NC2(c3ncc[nH]3)CC2)C1 10087,C(c1ccc(F)c(OC)c1)=CC(N1C2CC(NC(C(CCOC)C)=O)C2CC1)=O 10088,N1(C(C(C)NC(CC)=O)=O)CC2CC1C2NC(=O)C(C)=C1CCC1 10089,c1(CC(=O)NCCCCN(C(C(C)=C2CC2)=O)C)nc2nc(C)cc(C)n2n1 10090,C#CCC(CC(=O)NC1CCCCCC1)NC(c1cccc(C)c1C)=O 10091,C(C(C)(C)C(=O)NC(CNC(C1(c2ccccc2)CCCO1)=O)C1CCC1)SC 10092,c1(N(C)C)ccc(F)c(C(=O)NCCCCn2cc(-c3cccnc3F)nn2)c1 10093,N1(C(c2c(C)cc(SC)o2)=O)CCC(C)C(NC(=O)C=Cc2cn(C)cn2)C1C 10094,N1(C(CCC(=O)NC)=O)CCN(C(=O)C(C(C)C)OC)CC(C)(F)C1 10095,N1(C(c2c(C)noc2C2CC2)=O)CCCC(CC(=O)NC2(CC(C)=O)CC2)C1 10096,c1(C(N2CC(F)(COCC(=O)NC3CC(CF)C3)C2)=O)cccc(-n2cncn2)c1 10097,C1(C(=O)NC(CC)CNC(C2(OC(C)C)CCCC2)=O)CCC(F)(F)C1 10098,c1(CN2C(C(N3CCC(C(F)(F)F)C3)=O)CC(O)C2)cc([N+](=O)[O-])cc(Br)c1O 10099,Cc1ccc2nnc(C(=O)N(C)CCNC(C3(C)CCOC(C)C3)=O)n2c1 10100,N1(C(C#C)C)CCCN(C(C(=O)Nc2ccc(OC)cc2)C2CC(OC)C2)CC1 10101,C1(C#N)(CC(=O)N(CC(C(=O)N(CCCOCC)C)C)C)CCOCC1 10102,C(=O)(C(CC(C)C)NC)N(CCN(C(=O)C(O)C1CC1)Cc1ccccc1)CC 10103,C1(F)(CC(=O)N(CCCCNC(=O)CC2(CS(C)(=O)=O)CC2)C)CCCC1 10104,c1(-n2cc(C3(OC(C)C)CCC3)nn2)ccnc(Br)c1F.N12CCCC1C2=O 10105,N#CC1CN(C(c2ccc(CCO)cc2)=O)CCN1C(C1CCC(CO)CC1)=O 10106,CCCCC(O)CC(=O)NCC1CC1CNC(C1CCC(CC)O1)=O 10107,C1(NC(CC2(C)N(C(CC(=O)NCC)=O)CC2)=O)C2CCC1CC2 10108,C(C(F)(F)C(=O)NCCCOC1CCN(C(=O)CCc2ccsc2)CC1)OC 10109,N1(C(CCC2C(C)(C)C2)=O)CCN(CCNC(C2CC(=C3CCC3)C2)=O)CC1 10110,N1(C(c2ncoc2C2CC2)=O)CCCC(O)(CNC(C2(O)CCOCC2)=O)C1 10111,N1(C(Cn2c(C)ccn2)=O)CC2(C1)CN(C(=O)Cc1ccnc(F)c1)CC2CO 10112,c1(OC)ccc(-c2nc(C)c(C(C)NC3c4nnnn43)s2)cc1.C1(SC)CC1 10113,c1(OC)cc(C)cnc1C(=O)NC1(C(=O)O)CC(OC)C1 10114,N#Cc1c(F)cc(C(=O)NC2CC(CNC(=O)C3=COCCC3)C(O)C2)cc1F 10115,Cc1ccc(F)c(-c2ccc(CN(C3CC3C3CC3)C)cc2)n1 10116,C(C(C)(C)CCCc1ccccc1)N(C)C(N1CC(CC(F)F)C1)=O 10117,Cc1ccc(CNC(C2(C)CC2)=O)cc1.c1(CC(C)N)ccnc(O)c1 10118,N1(C(CC(CC)SC)=O)CCC2(CC(NC(c3csc(O)n3)=O)C2)C1 10119,C(=O)(C1=C(CCl)N(CC(C)C)C(=O)NC1c1ccc(Cn2cccn2)o1)OC 10120,C(=O)(C#CC1CCOC1)NCC1C(C(=O)NC2C(C)(C)C2(C)C)CC1 10121,C(=O)(C1=CN(C)S(=O)(=O)N=C1C)NC(CNC(C(C(CC)O)(C)C)=O)CC(C)C 10122,C(=O)(C(CO)NC(=O)C(c1cn(C)nn1)NC(c1cnn[nH]1)=O)N(C)C 10123,CCCC(C(=O)NCCCN(C)C(c1csc(SCCC)n1)C)OC 10124,N1(C(CC(=C)Br)=O)CC2CCCC2(NC(=O)CCc2ccccc2Cl)C1 10125,Cc1cc(P(C)(C)=O)oc1C(=O)NC(C)CNC(c1cc(C2CC2)cs1)=O 10126,N1(C(C2C(C)(C(=O)OCC)C2)=O)CCC2(C1)CN(C(c1n[nH]c(C)n1)=O)C2 10127,N1(C(C=C(COC)C)=O)CC2ON=C(CNC(c3csnc3Br)=O)C2C1 10128,C1(NC(CCC#CC)=O)CC2(NC(c3scnc3COC)=O)COC1C2 10129,C1(C)(CCNC(C(C)O)=O)CCN(C(c2ccc(-c3cccnc3)cc2)=O)C1 10130,c1(CSC)cccc(CN2CCC(CC(N3CCC(Br)C3)=O)C2)c1 10131,Cc1ccc2c(CCC(=O)N3CC(N(C(=O)CCCS(C)(=O)=O)C)C3)c[nH]c2c1 10132,C1(C)(NC(c2ccc(CNC(c3n(C=C)ncc3)=O)s2)=O)CC2(CCC2)C1 10133,C=C(C)CCC(=O)NC(C1CN(C(=O)C(CCC)c2cccc(Cl)c2)C1)C 10134,C1(N=[N+]=[N-])(C(=O)Nc2c(CC)nn(C)c2)CCN(C(=O)CSc2nc[nH]n2)C1 10135,N1(C(C(C)(C)n2cccn2)=O)CC2(C1)CN(C(=O)CC1CCCCC1)CC2CO 10136,C1(C(N2CC=C(C)C2)=O)(C(C)C)CCN(C(=O)CCC2CCC2)C1 10137,CC(C)CC(O)CNC(=O)CCCCN(C)C(C1(CO)CCCCO1)=O 10138,c1(C(N2CCCCC2C2CCCC2O)C(=O)NCC)cc(Br)ccc1F 10139,CC1(C)C(c2cccc(Cl)c2)CCN1C(c1nn(CC(F)(F)F)cc1Cl)=O 10140,c1(C(=O)NC2CC(NC(c3c(CC)nccn3)=O)C2)nc(C2CC2)ncc1Cl 10141,CN1CCCC1(C)C(=O)NCC12CC(NC(C3CCCS3(=O)=O)=O)(C1)C2 10142,C(=O)(C#CC1CCCO1)NCC(CC(C)C)NC(=O)CSc1nncn1C1CC1 10143,C1(C(=O)NCCCCNC(C(C)CN2CCOCC2)=O)Cc2ccc(F)cc2O1 10144,C1(c2ccccc2)(NC(CCN(CCCCC)C)=O)CCN(C(=O)CC2CC2)C1 10145,c1(C(=O)NCCCCCN(C(c2ccc(CC)nc2)=O)C)ccc(C)c(N)c1 10146,c1(C(N2CC(NC(C3(O)CCOC3)=O)CC(C)(C)C2)=O)cnnc2ccccc12 10147,C1(NC(c2c(C)nns2)=O)CCCN(C(=O)CC2CCN(C)C2)C1C 10148,c1(C(=O)NC(C2C3CNCC23)C(=O)OC)csc(Cl)c1OC 10149,c1(OC)ccc(O)cc1C(=O)NCC1CCCC(NC(C2CC(F)C2)=O)C1 10150,c1(C(N2CC(N(C(c3c(C)nccc3)=O)C)C(O)C2)=O)cc(C2CC2)nnc1O 10151,c1(CC(=O)N(C2CCN(C(c3c(CC)cco3)=O)C2)CC2CC2)cncnc1O 10152,n1(-c2cn(C)nc2)nc(OC(F)(F)F)nc1-c1cnco1 10153,CC(CCN(C(=O)CCC1OCCO1)C)NC(=O)Cc1nc[nH]n1 10154,Cc1cccc(N2CCC(NC(=O)CC3(C)CCOC3)C2=O)c1 10155,N1(C(c2cn(CCO)nn2)=O)CCC2CN(C(C3CC(C4CCC4)C3)=O)C2C1 10156,C1(C(=O)NOCC2CCCO2)(CC#C)CCN(C(=O)CCCC#N)C1 10157,c1(C(=O)NCC(CN(C(c2ncc(C)c(C)c2)=O)C)C)ccc2ccnn2c1 10158,C1(C(N2CC(OC)(CNC(=O)C(C)C3CCCC3)C2)=O)COC(=O)N1C 10159,N1(C(C2CC(SC)C2)=O)CC(NC(c2csnc2C)=O)CC12CCCC2 10160,CC(=O)CCCC(=O)N(CC(=O)NCC1CC(O)C1(C)C)C(C)C 10161,C1(NC(c2c(C(C)C)nns2)=O)CN(C(=O)C2=CSCCO2)CCC1CO 10162,N1(C(c2ncn(C)n2)=O)CC(NC(=O)C(F)(F)C2(O)CCC2)CC12CCCCC2 10163,CCC(C(=O)NCC1(CCNC(=O)Cc2ccncc2Cl)CC1)C(F)(F)F 10164,C12(NC(=O)COc3ccon3)CCCN(C(C3(CO)COC3)=O)CC1C2 10165,N1(C(CCC=CC)=O)CC2CC1C2C(N1C(C)CC1(C)C)=O 10166,C1(C2CN(C(=O)C(F)(F)C3(O)CCCC3)C2)(NC(c2ccc(CF)cc2)=O)CC1 10167,c1(C(=O)NC(c2cccc3cc[nH]c23)CC)cnn2cc(-c3nn[nH]n3)cnc12 10168,c1(C(N(CC(O)CNC(C2CCSC2)=O)C)=O)cc(P(C)(C)=O)cs1 10169,CC1CC(C(=O)NCCCOCCC(=O)NCC(C)(F)F)=NO1 10170,c1(C(=O)NCCCN(C(=O)CCN(CC(F)(F)F)C)C(C)C)cc(Br)c[nH]1 10171,c1(C(=O)NCCC(C)NC(C(C)OCC)=O)ccc(S(=O)(=O)C(F)F)cc1 10172,Cc1cccc2c(C(N3CC=CC3CNC(C34CCC(CO3)C4)=O)=O)n[nH]c12 10173,c1(C(=O)NC2CC(F)(CNC(C3(CC(F)F)CCC3)=O)C2)cc2cn[nH]c2cn1 10174,c1(C(=O)NCC2C(C)(C)C(NC(=O)COC3CCC3)C2)ccccc1[N+](=O)[O-] 10175,CC1C(=O)CC2CCC1N2Cc1ccc(C(C)(C)C)cc1 10176,Cn1cc(SCC(=O)NC2(CNC(=O)C(C)(c3cccs3)N(C)C)CCOC2)cn1 10177,c1(C(=O)NCC2(F)CC(CNC(C(F)=C(C)C)=O)C2)cccc(Br)c1C 10178,c1(C(N2C(CNC(C(C(C)C)C)=O)CC(O)C2)=O)cc(=O)n(C)cc1Br 10179,c1(NC(c2ccc(-c3ccc(Br)s3)s2)=O)ncccc1OCCF 10180,C(=O)(C(O)C1=CCCCC1)N1C(C2(NC(CC(=O)NCC)=O)CC2)CCC1 10181,CCC(C)(CS(C)(=O)=O)C(=O)NCC(O)CNC(=O)CNC(=O)NC 10182,c1(C(=O)NC2(CN(C(C(CC)OC)=O)C)CC2)cc2c(C#N)cccc2[nH]1 10183,N1(C(CSCC#C)=O)CC(C2CCCN(C(C3(CO)CCCO3)=O)C2)C1 10184,N1(C(Cc2c(C)nc[nH]2)=O)CCC(CO)C(NC(C2(C(C)C)CCC2)=O)C1 10185,CN1CCC(C(=O)NC2COCC2CNC(=O)Cc2cccnc2Cl)CC1=O 10186,c1(C(N(CCC(C)NC(=O)C(C)(C)C)C)=O)ccc2c(c1)OC(C)(C)OC2 10187,CC(C1OCCc2ccccc21)NCc1csc([N+](=O)[O-])c1 10188,O=C(C(CCC1CCC1)NC(C1CC=CC(O)C1)=O)NCc1ccc(O)nn1 10189,N1(C(Cc2c(C)scc2)=O)CCC(CC(=O)NCCCCCCO)C1(C)C 10190,C1(NC(C(C)Nc2cccnc2)=O)COCCN(C(C2C3COCC23)=O)C1 10191,N1(C(C2CCCC(C)(C)O2)=O)CC=CCC12CCOCC2 10192,C1(CNC(CNS(N)(=O)=O)=O)CC2(CCC2)CN1C(c1cccc(C2CC2)n1)=O 10193,n1(CCC)nccc1S(=O)(=O)NCc1nc(NC(C)=O)n(-c2ccccc2)n1 10194,N(C)(S(=O)(=O)N(C)CC1CC1)CC#C 10195,c1(C(C(=O)NCC=CCl)NC(CN(C)CC)=O)cnn(C)c1 10196,C1(NC(C(n2cc(-c3ccn(C4CC4)n3)nn2)C)=O)CCN(CC2CC2)CC1 10197,N1(C(C2C(C)(C)N(C(=O)CC3CC4(CC4)C3)CC2)=O)CCOCC2(CC2)C1 10198,C1(CNC(CN(C2CC2)CC)=O)CN(C(c2cscc2OC)=O)C2CC12 10199,C(N=c1[nH]c(N(CCCS(C)=O)C)nc2c1CCCCC2)c1ccc(SC)cc1 10200,C(=O)(CS(=O)(=O)CCO)NC1CCCC(NC(c2cncc(SCC)n2)=O)C1 10201,N1(C(C(COC)CC(C)C)=O)CC(C)OC2(CCN(C(=O)CCC(C)C)CC2)C1 10202,C1(C(N2CCN(C(CNC(C(C)C#N)=O)C)CC2)=O)CCCCC12CCC2 10203,c1(OC)ccc(NC(c2ncsc2C(C)C)=O)cc1C#N 10204,c1(NCCCC(C)NC(C(C(C)C)O)=O)ncnc2ccc(C(F)(F)F)cc12 10205,C(CC(C)C(=O)NC1CCC(F)(CNC(c2c[nH]c(C(F)(F)F)c2)=O)C1)OC 10206,Cc1nsc(NC(N2CC(F)CC2CO)=O)c1Cl 10207,C(CC(C)C(F)(F)F)NC(C1(CNC(C=CCC)=O)CCC1)=O 10208,C1(CNC(C(CC=C)NC(C)=O)=O)CC(C(=O)NCC2(N(C)C)CCC2)=NO1 10209,N1(C(C(C2CN(C(=O)CC3CC=CC3)C2)OC)=O)CC(OC)C(C)(C)C1 10210,C1(NC(C2C(CC)CCC2)=O)CC2(CCN(C(C3(C)CCN(C)CC3)=O)C2)C1 10211,C1(NC(C2(COC)CCOCC2)=O)CCN(C(c2ccsc2C)=O)CC1(C)C 10212,c1(C(N2CCC(O)(CNC(C3C(CCOC)C3)=O)C2)=O)ccc([N+](=O)[O-])o1 10213,C(=O)(C(C)(O)C(C)C)N(CCC(=O)NC1C2CCCC12)CC=C 10214,C=C(C)CCCC(=O)NCC1(O)CCCN(C(=O)C=CCOc2ccccc2)C1 10215,C1(NC(C(C)OCC)=O)CCN(C(=O)Cc2ccc(C(C)=O)s2)CC1(C)C 10216,CC(C)C(C(=O)NC(CNC(=O)Cn1cnnn1)C(C)(C)C)NC=O 10217,c1(CC)[nH]nc(C(=O)N(CC(=O)N(C2CCCCC2C)C)C)c1C 10218,N1(C(=O)N(C(C)(C)C)C)CCCC(C)(CCn2cc(CC(O)SCCCl)nn2)C1 10219,N1(C(=O)NCc2ncc(CC)o2)CCCCC1CCNC(C)=O 10220,c1(CNCc2ccc(OC)nc2Cl)cccc([N+](=O)[O-])c1.C12CCCCN1C2=O 10221,N1(C(C(=O)NCCOC(C(C)SCC)=O)C2CC2)CCC(OC(C)C)CC1 10222,CC(C(=O)NCc1cnsc1)F.C1CCCC2CN1C2 10223,Cc1ncc(NC(=O)NCCc2ccccc2Oc2ccc(Cl)c(Cl)c2)cc1Br 10224,C(=O)(C1CCc2ccccc21)NC1(C(=O)NC(C=C)CO)CC(CO)C1 10225,C1(C(=O)NC(c2ccns2)C)(CC)CCCN(C(c2cnn(C(F)F)c2)=O)C1 10226,C#CCCCCCC(=O)N1CCCC2(NC(C3CCOC3)=O)CC2C1 10227,Cc1cc(C(=O)Nc2ccc(NC(=O)CCn3ccnn3)c(C)c2)ncc1N 10228,c1(NC(C(CCC)C)C)ccc(S(=O)(=O)N(C2(CCO)CCSCC2)C)cc1Br 10229,c1(C(=O)NCCC2CCCN(C(C3CC(F)C3)=O)C2)nccc2n[nH]cc12 10230,c1(C(=O)NCCC(N)=O)cncc(CNC(C2CCC2(F)F)=O)c1 10231,N1(C(CC(C)OC)=O)CC2(CCN(C(=O)C(C)Sc3ccc(N)cc3)C2)C1 10232,c1(C(N2CCCSCC2C)C(=O)Nc2c(OC)cccc2)sc(C)c(Br)c1C 10233,C1(C#N)(NC(CSc2ccc(OC)cc2)=O)CCN(C(=O)CC2CCCCC2)C1 10234,C(=O)(C(C)(Cc1ccccc1F)NC(C1CC=CCO1)=O)OC 10235,c1(NC(=O)NCc2cccc(-c3cccc(OC)n3)c2)ccc2sc(O)nc2c1 10236,c1(C(N2C(CNC(CNS(N)(=O)=O)=O)CC(O)C2)=O)cnn2c1CCC2 10237,O=C1CC2(CCCN(C(=O)C3=NOC(CO)C3)CC2)CN1 10238,CC(CN(C)C)C(=O)N1CCCC1C(C)NC(=O)N(C)C 10239,C(=O)(C(CNC(=O)CN1CCCC1=O)C(C)C)N1CCC(C(=O)NC)CC1 10240,C1(CC(=O)NC(C)C(=O)Nc2cnn[nH]2)CN(C(=O)OC(C)(C)C)CC1C 10241,CCCC(CCC)CC(=O)NC1CN(C(C2CCCOCC2)=O)CC1OC 10242,C1C2c3ccccc3CN2C(=O)CC(=O)N1.C(c1cncs1)=CCC(C)C=O.OC 10243,c1(N(C2CCN(C(c3cnc(SC)s3)=O)C2)C)ncnc2sc(C(F)(F)F)nc12 10244,S(=O)(=O)(c1ccc(CC(=O)NCC2CCCN2C(=O)C(C)C(C)O)cc1)NCC 10245,N1(C(=O)OC(C)(C)C)CC2(C(=O)N(C(c3cncn3C)COC(F)F)CCl)OC2C1 10246,n1(CCNC2C(C(N3CCC(C(CC)CC)C3)=O)C2(C)C)ncccc1=O 10247,c1(C(=O)NC2CCN(C(C(C)SCC)=O)CC(O)C2)cnn2cc(OC)ccc12 10248,N1(C(C(C)NC(N)=O)=O)CCN(C)C(CNC(c2nsnc2O)=O)C1 10249,C1(N(C(C(=O)Nc2ccccc2)=O)CCCO)CC2CC1CN2 10250,c1(C(=O)OCC)ccccc1NC(C1CC1CNC(=O)CCc1ccn(C)c1)=O 10251,CC(CNC(C1(F)CCN(C(c2ccc(Cl)cn2)=O)CC1)=O)CC(F)(F)F 10252,C1(C(=O)NCC(CNC(c2c(C)n[nH]c2)=O)C)CCCN(CC(C)C)C1 10253,c1(N(C)CC2CCN(C(C3N(C(CCC)=O)CCCC3)=O)CC2)nnc(C)c(C)n1 10254,c1(NC(C2CCC(NC(C3N(C)CCCC3)=O)C2)=O)ccc(O)c(Br)c1 10255,CN1CCCC1C=CC(=O)NC1(C(=O)N(C2CSC2)C)CC(F)C1 10256,C12(COC)CCC1CN(N1C(C=O)CC1)C2.c1(C=O)ccc(CO)s1 10257,C1(Nc2nccc(OC)n2)(CO)CCN(C(C)=O)CC1.C12(CCCC1)C(=O)N2 10258,N1(C(CC2(N(C)C)CC2)=O)CC(NC(=O)Cn2cc(Cl)cn2)C(C(F)F)C1 10259,C1(OCC)CC(NC(=O)C(=O)NCCOS(=O)(=O)c2cccs2)C12CCCC2 10260,c1(OC)nsc(OC)c1C(C)NC(C1(n2cc(F)cn2)CC1)=O 10261,C1(C(=O)NCC(C)CNC(=O)Cn2nccn2)CC(O)c2ccccc2O1 10262,C12(OC)CCCN(C1)C2c1n(CCCCCC)nnn1.C(C)(CC(C)C)OC 10263,C1(C(=O)OC)CCOC1C(=O)NCCN(C)C(C1CC(C(C)C)C1)=O 10264,C(CCCC(=O)N1CC2C(CNC(=O)C(c3ccc(Cl)s3)=O)C2C1)SC 10265,CCS(=O)(=O)CC(=O)NC1(CO)CCN(C(c2cccc(OC)c2OC)=O)C1 10266,c1(C(N2CCCC(CNC(C(C)(C)OCC)=O)C2)=O)cc(Cl)c(OC)cc1C 10267,C(=O)(C(C)(C)CS(C)(=O)=O)NCCCC(C)NC(=O)C(O)CC(N)=O 10268,C(=O)(CC(C(C)C)NC)N1C(N(C(=O)C(=O)NCCOC(C)C)CC)CCC1 10269,C(=O)(C(C(C)C)NC(=O)CNC1C(C)C1C)OC(C)CC 10270,Cc1cnc(Cl)[nH]c1=NCC=Cc1ccc(OCC2CCCCC2)cc1 10271,N1(C(c2c(Cl)ncc(C)c2)=O)CC2CCN(C(c3c(Br)cnn3C)=O)C2C1 10272,c1(C(C)C)cc(C(=O)NCCNC(=O)CCC(C)C#N)ccc1F 10273,N1(C(C2CCN(C(=O)CCc3ccccc3)CC2)=O)CCOCC2(CCC2)C1 10274,c1(C(=O)NCC(CN(C(c2c(C)noc2N)=O)C)C)cc(Cl)ccc1Cl 10275,N1(C(CCC2C(C)C2)=O)C2CCC1CN(C(c1csnn1)=O)C2 10276,Cc1cc(C(=O)NCC2CN(C(=O)COCCF)CC2C)c2c(C)nn(C)c2n1 10277,c1(C(=O)NCC(C2N(C(C(CC)CC)=O)CCCC2)(C)C)cnc2ccnn2c1 10278,N1(C(=O)CCN(C(c2nsnc2O)=O)CC2CC2)CC23CCC2(COC3)C1 10279,c1(NC(C2(C)CCN(C(c3ccc(CF)cc3)=O)C2)=O)ccc(F)c(O)c1 10280,Cc1nn2c(C(N3CC4CC4(NC(C4(N5CCCC5)CCC4)=O)C3)=O)c(C)nc2s1 10281,CCC(Cc1ccccc1C)C(=O)NCC(C(C)C)NC(=O)CC1CC=CC1 10282,C(=O)(C(C(=O)N1CCCC(CNC(=O)CC(NC(=O)NC)CC)C1)OC)OCC 10283,C(=O)(CC(C)C(F)(F)F)NCC(CNC(c1ccc(NC)cc1Cl)=O)OC 10284,C1(CCNC(CCC#CC)=O)CN(C(C2CC3CCC3C2)=O)CCS1(=O)=O 10285,C1(C(=O)NC2(CCC)CC2)C(C2CC2)CCN1C(=O)COCCCF 10286,C1(C(N2CCN(C(c3cc(Cl)cnn3)=O)C(CO)C2)=O)CCCNS1(=O)=O 10287,N1(C(CC2(C(=C)F)CCC2)=O)CCC(C(=O)NCC(Cl)C(C)(F)F)C(C)C1 10288,N1(S(CC)(=O)=O)CCC(C(=O)NCC2CN(C(=O)C=CCOC)CC2O)CC1 10289,C(=O)(CCC(=O)NCCCCCCNC(C1CC1(Br)Br)=O)NCC 10290,C1(NC(CC2CN(C(C)=O)C2)=O)CN(C(c2cc(Cl)ccn2)=O)C2(CCOC2)C1 10291,c1(OC)ccc(-c2cn(CC3CN(C(C4(F)CC=CC4)=O)CCO3)nn2)cc1Br 10292,C1(C(=O)OCC2C(Cl)(Cl)C23CC3)CNC(=O)CN1C(=O)NC(C)(C)C 10293,C#Cc1ccc(C(N2CCCC2CCC(N2CCOCCC2C(N)=O)=O)=O)cc1 10294,c1(C(C)C(N2CCC(CNC(=O)Cc3cccnc3)C2)=O)ccc2c(c1)CCO2 10295,C(=O)(C(CC(C)C)C(C)C)NCC1(OC)CN(C(c2cnc3n2CCC3)=O)C1 10296,Cc1c(CN2CC3(CCN3C(c3cc(Cl)cnc3Cl)=O)C2)[nH]c2ccccc12 10297,N1(CC)CCCCC1C(=O)NC(C)C(=O)O.C12CCN(C1)C2=O 10298,C1(CC#N)CN(Cc2cccc(-c3ccccc3)c2)CCN1C(C1CC1F)=O 10299,Cc1ccc(C(=O)NCC(=O)NCC(C2CC2)NC(=O)C=CSc2nc[nH]n2)s1 10300,N1(C(c2cnc(C)c(N)c2)=O)CCCC12CCN(C(=O)C(C)CC(C)(F)F)C2 10301,CC(N=[N+]=[N-])C(=O)N1CC(C(=O)NCCC2COCC2O)C(C)C1 10302,N1(C(c2ccn(CCCC)n2)=O)CC(NC(=O)CN2CCCCCC2)CC(F)C1 10303,c1(C(=O)NC2(CNC(C3=CCC(C)(C)CC3)=O)CC2)cc(Cl)cc2c1NCCC2 10304,N1(C(c2cc(CC)nc(O)c2)=O)CC2(CCN(C(=O)C(C)NC(=O)NC)C2)C1 10305,C1(CNC(c2c(C(=O)OCC)c[nH]c2)=O)C(C)CCCN1C(=O)CCC(C)(F)F 10306,c12cnn3c(cccc13)NC2=O.C1(C(=O)O)(C(=O)O)C2CCC12 10307,C1(C(N2CCC(CCOC)(NC(CC=CC)=O)C2)=O)CC2COCC2C1 10308,C1(C(=O)NCC(CCC)OCC)CCC2CCC1N2C(c1ccccn1)=O 10309,N1(C(Cc2c(C)oc(-c3ccsc3)n2)=O)CCc2nncn2CC1 10310,CC(C)C(C(=O)NC1(C)CN(C(C2CCC(=O)C2)=O)C1)c1cccc(Cl)c1 10311,c1(C(N(C(CNC(CCc2cc(C)[nH]n2)=O)C2CC2)C)=O)nc(C)n(C)c1C 10312,c1(CC)cc(C(=O)NC2CN(C(=O)CO)CC2SC)nn1CCO 10313,c1(OC)ccc(CNCC(N)C(C)C)cc1Cl 10314,C12(CNC(c3cncc(COC)c3)=O)CCC(CC1)CN2C(=O)CC1CCC1 10315,c1(CC)ccoc1C(=O)N(CCNC(c1ccc(CS(C)(=O)=O)o1)=O)CC1CC1 10316,c1(CNCC2(C(=O)O)CCSC2)ncnc(O)c1F 10317,N1(C(C(C2CCCO2)SC)=O)CCC(N(C(=O)CCOC2CCC2)CC2CC2)CC1 10318,N1(C(c2cnc(Br)s2)C(=O)NCC=C)CCC(C)(O)C(C)(O)C1 10319,N1(C(c2nccc(C)c2O)=O)CCC2(CCC2)C(NC(C2CCCSC2)=O)C1 10320,C1(CNC(CC=C(C)C)=O)CCC(n2cc(CC3(O)COC3)nn2)CC1 10321,S(=O)(=O)(c1ccc(NC2(C(=O)O)COC(C)(C)C2)cn1)NC(=O)OC(C)(C)C 10322,N1(C(CCCCCOC)=O)CC(CNC(C2(CF)CC2)=O)CC12CCC2 10323,N1(C(CC2C(=O)NC(=N)S2)=O)CC2=C(C1)CN(C(C13C4C5C1C1C3C4C51CO)=O)C2 10324,c1(C(=O)NC(CC2(CC)CCC2)=O)cc(CN2CCCC(NC(C)C)C2)ccn1 10325,C(=O)(C(C)(C)C(C)(F)F)NC1C(C(C)C)N(C(=O)CC2CCOCC2)CC1 10326,Cn1c(NC(C2CC2NC(=O)Nc2cccc(C#N)c2)=O)cc2cc(Cl)ccc12 10327,C(=O)(CCCC(=O)N1CCC(C(F)(F)F)C(OC)C1)NCCC 10328,C1(NC(c2c(CC)nc(C)nc2)=O)CN(C(=O)Cc2ccnn2C)CC12CCC2 10329,N1(C(CN(S(C)(=O)=O)C)=O)CCN(C)c2ccc(NC(=O)OC(C)(C)C)cc21 10330,Cc1c(C(=O)N(C)CCN(C)C(c2occc2C2CC2)=O)ccn1CC1CC1 10331,C(=O)(N=S(=O)(c1ccc(F)cc1)C(F)F)c1cccc(N=S(C)(C)=O)c1 10332,C1(CC=C)(NC(c2csc(CC)n2)=O)CN(C(=O)C(F)CC2CCCC2)C1 10333,N1(c2nc(OC)nc(C)c2)CCOC2(CCCN(C(C3CCCCC3C)=O)C2)C1 10334,Cc1ccc(C(=O)NCC(N2CCN(C(=O)C3=NOCC3)CC2)C)c(F)c1 10335,C1(CCOC)(NC(=O)C=C(C)C(C)C)CCN(C(=O)CN2CCS(=O)CC2)C1 10336,C12(CNC(C(C)C3CCCC3)=O)CC(CO1)N(C(=O)Cc1ccc(F)c(Cl)c1)C2 10337,c1(C(=O)NC(CCCNC(c2n(C(C)C)ncc2)=O)C)nnn2c1C(=O)NCC2 10338,c1(C(C(=O)NCc2cn(CCCOC)nc2)O)cccc(Cl)c1 10339,C(=O)(CCCCCc1ccccc1)NC1C(CNC(c2c(CC)cc[nH]2)=O)C1 10340,N1(C(C2CC(N(C)C(C34CC(CO)(C3)C4)=O)C2)=O)CCC([N+](=O)[O-])CC1 10341,C(=O)(CCCCCC#N)N1CC(C(=O)NCC(C)C2CCC2)N(C)CC1 10342,C1(CNC(CS(CC)=O)=O)COCCN(C(C2CC(N3CCCC3)C2)=O)C1 10343,C(C(CC(=O)N(C1CCSC1)C)NC(=O)C=Cc1cc(C)no1)OC 10344,C1(NC(c2ccc(CC)c(Cl)c2)=O)COC2C(NC(=O)CC(=O)N(C)C)COC12 10345,C(=O)(CCC(C)(C)C)N1CC(C)C(CNC(c2cn(CCCF)nn2)=O)C1 10346,c1(C(=O)NC2CC2NC(C2COC3(CCC3)C2)=O)cnc2cc[nH]c2c1 10347,N12CC3CCC3(C1)C2=O.Cc1cc(C(=O)Nc2ncc(C3OCCO3)s2)nn1C 10348,N(C1CCCn2ccnc21)C(C(CCNC(c1c(C)cn(C)n1)=O)O)=O 10349,c1(C(=O)NC(CC=C)CNC(=O)C=Cc2scnc2C)cccc(S(C)=O)c1 10350,N1(C(C(CSC)C)=O)CCC(O)(CNC(c2c(C)coc2C)=O)C1 10351,Cc1nsc(C)c1C(=O)NCC1CC(C)N(C(=O)Cc2ccc(C(N)=O)nc2)C1 10352,Cn1nnc(C(=O)NCCOCCNC(=O)CCCc2ccccc2)n1 10353,C12(NC(c3c(CC)ocn3)=O)CCN(C(c3cc(C(C)(C)C)no3)=O)CCC1C2 10354,N1(C(CSCCC(C)C)=O)CCCC2(NC(c3cncc4sccc34)=O)CC2C1 10355,c1(N2CCCC(N(C(COc3cccc(OC)c3)=O)C)C2)ccc2nnnn2n1 10356,CC12CCC(C(N3CCOC(CNC(=O)CSC4CC4)C3)=O)(CO1)C2 10357,C1(CNC(c2scc(C)c2)=O)CC2(CO1)CN(C(C1(C)CCCNS1(=O)=O)=O)C2 10358,c1(C(N2CC(C(N)=O)(CNC(CC(=C)C)=O)C2)=O)cccc2c1OC(C)C2 10359,c1(C(N2CCCCC(NC(c3cc(OC)no3)=O)C2)=O)cnc2c(n1)CCCC2 10360,c1(C(N(C)CC2N(C(C(C(CC)C)O)=O)CC(F)C2)=O)cc(C)cc(C)c1C 10361,N1(C(C2N(C(C3C(C)C4CCC3C4)=O)CC(F)(F)C2)=O)CC(=O)N2CCCC2C1 10362,c1(C(=O)NC2(C)CC(OCC)C2)ccc(-c2ccccc2)c(C)n1 10363,C1(CNC(CN(C)C2CC2)=O)CCCC(NC(C2(O)CCOCC2)=O)C1 10364,C(=O)(C(C)C(C)S(C)(=O)=O)N1CC2C(CNC(CCCCC(C)C)=O)C2C1 10365,N(C1CCc2cccnc21)C(C1N(C)CCN(C(C2N(C)CCCCC2)=O)C1)=O 10366,C(=O)(NN=Cc1cccnc1Br)c1nnc(-c2c(C)ccc(F)c2)s1 10367,N1(C(c2c(C)ncnc2)=O)CCC2(CC1)COC(CNC(=O)C(C)C(C)C)C2 10368,C(=O)(N1CCCc2nccn21)c1ccc(CNC(=O)C=CCN2CCC2)cn1 10369,c1(C(=O)NC2(CNC(c3n[nH]c(C)c3F)=O)CCOC2)ccnc2ccsc12 10370,N1(C(c2cncc(C=C)c2)=O)CC2(C(=O)NCC3CCOC3)CCC1CC2 10371,c1(OC)cc(OC)cc(C(=O)NC2CCCC2CNC(C2CC(OC)C2)=O)c1 10372,C1(NC(C(C(C)C)SC)=O)CCC(C)N(C(=O)CC2(O)CCCCC2)C1 10373,CC#CCC(C(=O)NC(COC)C1(C)CC1)NC(=O)Cc1cnn(C)c1 10374,Nc1cc(C(=O)NCC2(NC(=O)CCn3ccnn3)CC3CCC2C3)cc(F)c1 10375,c1(OCCC)cccc(C(c2nnnn2C)N(C2CCC2)C2CC2)c1 10376,CC1(C2CCCN(C(C3CC34CC(NC(=O)COc3cccnc3)C4)=O)C2)CC1 10377,c1(CC)cc(N)ccc1C(=O)NC(C)(C)CNC(C1(C(F)(F)CC)CC1)=O 10378,N1(C(c2c(C)nn(C3CCC3)c2)=O)CCC2(CCC2)C(NC(C2CC(O)C2)=O)C1 10379,n1(CC(=O)NCCC(C)NC(=O)CCOC2CCOC2)cnccc1=O 10380,c1(OC)ccnc(O)c1C(=O)NC1CCCCN(C(C2Cc3nncn3C2)=O)C1 10381,N1(C(c2c(C)ccc(NC(COC)=O)c2)=O)CC(C)N(C(=O)CCF)C(C)C1 10382,N1(C(COCC(C)C)=O)CCC(N(C)C(C2CC3(CC(=O)C3)C2)=O)C(C)C1 10383,CC(CC1CCC1)C(=O)NCC1(NC(c2cnnn2C)=O)CCCC1 10384,C1(C(C(C)C)NC(Cc2nnc(C)o2)=O)CCN(C(C2(O)COC2)=O)CC1 10385,C(=O)(C1=CC2CCC1C2)NC1CC(NC(c2cn(CC(=O)N(C)C)nn2)=O)C1 10386,S(=O)(=O)(c1ccc(OC)cc1)NCCCc1cccc(OC)c1 10387,c1(N2CCC(N(C(C(COC(C)C)(C)C)=O)C)C2)nc(O)c2ccc(Cl)cc2n1 10388,c1(C2(C(=O)NCCN(CCC)C(C3CC3[N+](=O)[O-])=O)CC2)ccccc1 10389,C1(C(=O)NC2CC(NC(C3CCCC4(CCC4)C3)=O)C2)CCC2(CCCO2)CC1 10390,N1(C2CN(C(C(C)NC(c3ccccc3)=O)=O)C2)CCC(NC(=O)CCF)CC1 10391,c1(OC)c(C(N2CC(C)(NC(=O)CCCCc3cnc[nH]3)C2)=O)c(C)nn1C 10392,C1(NC(C23CC(C)C2C3)=O)CN(C(c2ccc(CS(C)(=O)=O)o2)=O)C(C)(C)C1 10393,N1(C(C)C)C(=O)CCC1C(=O)N(C1CCN(C(=O)CC2(C3CC3)CC2)C1)C 10394,c1(CC(=O)NC2(CC=C)CCN(c3nccn4nnnc34)C2)ccc2c[nH]nc2c1 10395,C(=O)(C(C)(C)CF)NC(C)C(c1ccccc1)NC(c1cnc(N)cn1)=O 10396,Cn1cnc2nc(N3CC=CC(NC(c4cc(C5CCCC5)[nH]n4)=O)C3)ncc12 10397,CC(C)(C)C(O)CCC(=O)NCC1CN(C(C2CC2C(F)(F)F)=O)C1 10398,c1(SC)ccccc1C(=O)NC(C)CC1CN(C(=O)Cc2[nH]nnc2C2CC2)C1 10399,Cn1ccc2nc(N3CCCC(S(=O)(=O)N(C)C)C3)ncc12 10400,c1(SCC(=O)N(C2CCCCCC2)C)ccc2c(c1)CCCN2 10401,c1(CC(=O)NC2C3CN(C(C(CC)=CC)=O)CC2C3)ccc2nsnc2c1 10402,CCC(C)(C)CCCC(=O)N1CCC(N(C)C(C2CC3CCC3C2)=O)C1 10403,C#CCC(C(=O)NC1CCN(C(N)=O)CC1)NC(=O)CC1CCCC1O 10404,c1(OC)cnc(C(=O)N(C)CCN(C)C(c2n[nH]cc2CC(C)C)=O)c(OC)n1 10405,C(C#Cc1ccccc1)N1CCN(C(=O)CC2(O)CCOC2)CC1 10406,C1(CCOCCNC(=O)CC2CCCO2)CN(C(=O)C(=O)N(C)C)CCC1(F)F 10407,c1(C(=O)NCC2C(NC(c3ccn(COC)n3)=O)C2)cccc2c1OCC2C 10408,CC(C)CC(=O)C(=O)N(CCCCC(=O)NC(C)CCCCO)C 10409,N1(C(CCNC(C)=O)=O)CCC2(CC1)OCCCC2NC(=O)CSc1ccon1 10410,C1(CNC(c2cc(C)on2)=O)C2CN(C(=O)C(C)(C)N3CCOCC3)CC12 10411,C1(OC)CCC12CC(C(=O)NCCC1CCN(C(c3cnc(=N)[nH]c3)=O)CC1)C2 10412,C(CCF)(C(=O)NC(C)Cc1ccccn1)NC(c1c(C)csn1)=O 10413,C#CCCCCCCC(=O)N(C(C(=O)NCCC1CCC(=O)N1)C1CC1)C 10414,C(=O)(CC(C)C(F)(F)F)NCCCC(C)NC(c1onc(CC)c1C)=O 10415,N1(C(CC2(COC)CC2)=O)CC(NC(c2ccc(-c3csnn3)cc2)=O)C(O)C1 10416,N1(C(C(CC2CC2)NC(c2nccc(OC)c2)=O)=O)CCOC(C2(C)N=N2)C1 10417,C1(NC(C23CC(NC(COC4(C#C)COC4)=O)(C2)C3)=O)CCNC(=O)C1 10418,C(c1ccc(CN(C)Cc2cc(Br)ccc2Cl)cc1)=CC(=O)OC 10419,CC(C(=O)NCCOCCOCCNC(=O)C=Cc1ncc[nH]1)C(C)O 10420,CCCCS(=O)(=O)CC(=O)NCC1(C2CC2)CCN(C(C2CCS(=O)(=O)C2)=O)C1 10421,c1(CN2CCC(C#N)(C(C)C)C2)cc(Br)cc(F)c1O 10422,S(=O)(=O)(c1ccc(C(N2CC(CNC(=O)C(C)C#N)C(C)C2)=O)cc1)NC(C)C 10423,CC1CCCC(CC(=O)NCCCCCNC(c2csc(C#N)c2)=O)C1 10424,N1(c2nccc(OC)n2)CCC2(CC1)CC2NCc1ccn(-c2ccccc2)n1 10425,C1(CNC(C=C(CC)C)=O)CC2CCC1N2C(=O)CCn1cnccc1=O 10426,C1(C(=O)NC2(CC(=O)NCC3(C#N)CCCC3)CCCCC2)CC(C2CC2)=NO1 10427,C1(O)(CCNC(C(C)C#N)=O)CCN(C(c2cc(C(N)=O)n(C)n2)=O)CC1 10428,c1(C(=O)NCC(C)(CO)NC(CC(CC)C(F)F)=O)c(F)ccc2occc12 10429,c1(CNC(C2=NOC(C)(C)C2)=O)ccc2c(c1)CN(C(C13CC(CO)(C1)C3)=O)C2 10430,C(=O)(C(CC(C)C)C(C)C)N1C2(C(=O)NC(c3cn(CC)nc3)C)CC(C1)C2 10431,C(=O)(C(CCS(C)(=O)=O)OC)NC1C(NC(c2n(CC)cc(Cl)c2)=O)CC1 10432,C1(C(Cc2nnnn2C)NC(c2ncnn2C)CC)CCC(F)(F)CC1 10433,C(CN=c1cc(NCC2CCCC2)nc(COC)[nH]1)SCCCNS(CC)(=O)=O 10434,C12(NC(CNC(N)=O)=O)CC1CN(C(=O)CC(F)(F)Cl)C2 10435,c1(OCC(=O)NCC2CN(c3nnc(C(F)F)s3)CCO2)ccc(Cl)cc1 10436,N1(C(=O)NCC2CCSCC2)CCN(c2ccc(F)cc2F)C(=O)C1 10437,C1(C2(O)CCN(C(=O)C(C)C(C)(C)C)CC2)(NC(CCc2scc(C)n2)=O)CC1 10438,N1(C(C(CNC(C2CCC(=O)N2)=O)CC2CC2)=O)CCSC2(CCC2)C1 10439,C(=O)(C(C(=O)N1CCC(N2CCC3CCOC3C2)O1)C(C)C)OC 10440,CC1COC(C)CN1C(c1ccc(Cl)s1)C(=O)NCC1CC1 10441,C=C(Cl)C(C)(C)C(=O)N1CC2CC(NC(C3(F)CCOC3)=O)C1C2 10442,C1(C(N(CCCO)CCC)=O)CCCC1CNC(c1c[nH]cc1C)=O 10443,C#CCC(CC(=O)Nc1ccc(F)nc1)NC(C1(CC(C)C)CCC1)=O 10444,C(C(CNC(N1CCOC(C)(c2ccccc2)C1)=O)C(F)(F)F)OC 10445,c1(C(=O)NC2CC2CNC(C2CC3COCC3C2)=O)ccc([N+](=O)[O-])cc1Cl 10446,C1(C(=O)NC2CN(C(CCc3n(C)ccn3)=O)CC2O)CNC(=O)CC12CCC2 10447,Cc1cc(C(N2CC3CCN(C(=O)COC4CCOC4)C3C2)=O)c2[nH]cnc2c1 10448,N1(CC=CC)C(=O)CCC1CC(=O)NC1CN(C(=O)Cn2cc(C(C)=O)nn2)C1 10449,c1(C(=O)NCC2C(NC(C(c3nccc(C)c3)(C)C)=O)CC2)cc(Cl)ccc1N 10450,C(C(=O)N(C1CCC(NC(=O)CC(C)NC(N)=O)CC1)C)(C(C)C)OC 10451,N1(CCNC(C2CCC(n3cc(CN(C4CC4)CCl)nn3)C2)=O)CCC(O)C1 10452,c1(C(=O)NCC2N(C(CCCOC)=O)CCC2C)ccc2c(c1)CCS2(=O)=O 10453,c1(CC)cnn2ccc(C(N3CCC3CNC(=O)Cc3c[nH]nc3O)=O)nc12 10454,c1(C(N2CC3(CC(NC(=O)C=C4CCSCC4)C3)C2)=O)cnc2scnc2c1 10455,N1(C(=O)C2=NOCC2)CC2CN(C(C3C4C=CC(C4)C3CO)=O)CC(C1)O2 10456,Cc1cnc(C(=O)NCc2cccc(NC(=O)C(CC#N)c3ccccc3)c2)nc1 10457,C#Cc1ccc(C(=O)N2CCC(C(=O)N(CC(O)CN(C)C)C)O2)cc1 10458,c1(NC(C(c2cncc(Cl)c2)N(C2CSC2)C)=O)ccc(OCC(N)=O)cc1 10459,N1(C(CCC2CCC(NC(=O)C3=NOCC3)C2)=O)CCCCC(CO)C1 10460,N1(C(C(CCC)CCC)=O)CC2(C1)CN(C(C1CCC(NC)CC1)=O)CCO2 10461,CC1(CNC(C2(c3ccccc3)CC3(CC3)C2)=O)CCCN1C(c1ccsn1)=O 10462,C(CCCCCNC(=O)C(C1CCC(=O)N1)C)n1cc(C(C)OCC)nn1 10463,C(CN=c1nc(OC)cc[nH]1)C1CCC(NC(Cc2cc(OC)nc(C)c2)=O)C1 10464,Cc1nc(C(N2CC3CC2C3NC(=O)CC2(C)CCCO2)=O)cn1C 10465,N1(C(C)C(=O)NCc2ccncc2)CCN2C(C)COCC2C1 10466,c1(C(N(CC(CC)NC(C2C3CCCC23)=O)CC)=O)csc(-c2ccccc2)n1 10467,C(=O)(CCC(C)(C)F)NC1CCN(C(c2c(C(C)C)[nH]cc2)=O)CC1 10468,C(=O)(C(O)CC(C)C)N1C(COC)(CNC(=O)C(C)=C2CC2)CCC1 10469,C1(CCC(C)C)CCN(C(=NCCCCC(F)(F)F)NCCCF)C1 10470,Cc1cc(NC(=O)CCC(C)NC(=O)CCCN(C)C)cc(CO)c1 10471,C(=O)(C(CC(C)C)C(N)=O)NC(CC)CNC(c1sc(F)cc1Cl)=O 10472,C=CCC(CNC(c1cn2c(n1)CCC2)=O)C(=O)NC(CN(C)C)CO 10473,C(=O)(C(C)C1=CCCC1)NCCCN(C(=O)CCC(=O)c1ccccc1)C(C)C 10474,C1(CC)CCN(C(=O)C(C#N)C(C)C)C(C(N2CC(F)(F)C2C2CC2)=O)C1 10475,C1(CNC(C(C)=CC)=O)CCN(C(C2CCn3cc(C)nc3C2)=O)CCC1(F)F 10476,Cc1cccc(OCC(=O)NCC(C)N(C(=O)C(F)C2CCOC2)C)c1 10477,c1(C(c2nnnn2C2CC2)(CC)NCC2(C)CC=CC2)cc(OC)c(OC)c(Cl)c1 10478,Cc1ncc(CCNC(=O)C(C2CCN(C(c3csc(C)n3)=O)C2)C)s1 10479,c1(OCC(=O)N(C)CC2(O)CN(C(c3ccc(F)cc3)=O)C2)cncc(Cl)n1 10480,N1(C(C(C)(C)O)=O)C2CC1CN(C(C1(c3ccccc3F)CC1)=O)C2 10481,c1(OC)ccc2c(c1)C(C(=O)NC1(C)CN(C(=O)CCOC3CCCC3)C1)CC2 10482,N1(CC23CC(CF)(OC2)C3)CCC(N=c2nc(O)c3ccccc3[nH]2)C1 10483,C1(CNC(c2c(OC)n[nH]c2)=O)CN(C(C2(F)CC=CCC2)=O)CCN1C 10484,C(c1ccncn1)=CC(=O)NC1C(NC(CNS(NC)(=O)=O)=O)CC1 10485,c1(CNC(CC2(CSC)CC2)=O)cn(CC(N2CC(C(C)O)C2)=O)nn1 10486,C(=O)(C1(C)CCn2ccnc21)NCC(C)CN(C)C(c1csnc1Cl)=O 10487,C1(CC)CCOCCN1C(=O)CC(C1CC1)NC(c1cc(C)no1)=O 10488,C(=O)(CCCS(C)(=O)=O)N1CC2C(CNC(c3snc(C)c3N)=O)C2C1 10489,C=CC1(O)CCN(C(=O)Cc2ccc(F)cc2I)C1 10490,c1(C(=O)NCC2(O)CCN(C(Cc3n(C)nnc3)=O)C2)c2c(nn1C)CCSC2 10491,c1(C(=O)NCCCC(=O)N2CCC(c3nc[nH]n3)C2)ccc([N+](=O)[O-])o1 10492,Cc1cc(C(=O)NC2CC(NC(=O)CC3CCC3)C23CCC3)cc(Cl)c1 10493,C1(C(=O)NCC(CNC(C2(CSC)CCC2)=O)CO)CCC(C)(C)C1 10494,C1(C(=O)NC2C3CN(C(C4CC(=O)NC4)=O)CC32)CCc2nnnn2C1 10495,Cc1cc(=NCC(C)CNC(=O)C=C2CCSCC2)[nH]c(CO)n1 10496,C(=O)(C(C)S(=O)(=O)CCC)NCC(CC=C)NC(c1nc2cc(F)ccc2s1)=O 10497,N1(C(C)=O)CC=CC(N(C2CCCN2S(C)(=O)=O)C(=O)Cc2cccs2)C1 10498,C1(NC(=O)NCC2CC(C)OC2)(Cn2cc(C(N)=O)nn2)CC2(CCC2)C1 10499,Cc1cccc(C(=O)NCC2(CNC(C3(C(F)F)CCCO3)=O)CC23CCC3)n1 10500,C#Cc1cnc(CC(N2CCOCCC2C(=O)NCCC(=O)NC)=O)c(C)c1 10501,C1(CC(=O)NC2CN(C(=O)CCc3nncs3)C2)COC(=O)C1 10502,C(c1ccc(CN2CCCC2=O)o1)=CC(N1C(CNC(C(CC)=CC)=O)CC1)=O 10503,C(=O)(C1=CCC(C)(C)CC1)NC1(CNC(CC(CC)C2CCC2)=O)CCCCC1 10504,c1(NC(N(c2c(C)ccc(C)c2)CCC#N)=O)nc2cccnc2s1 10505,c1(CC)cncc(C(=O)NCC(CCOC)NC(C2(C(=O)NC)CCC2)=O)c1 10506,C(=O)(CC(O)CNC(=O)Cc1cccnc1O)N(C1CCC(C)(C)C1)C 10507,c1(C(=O)OC)cccc(F)c1NC(C1C2CCC(C2)N1c1ncc(Br)cn1)=O 10508,c1(C(N(CCN(C)C(c2csc(C3CC3)n2)=O)C)=O)c(N)ccc(F)c1F 10509,c1(C(N(C(C)CNC(=O)CC2(C)CC2)C)=O)cc(F)c(F)c(O)c1F 10510,C(CCC(C)(C)C(=O)Nc1ccc2c(c1)OCO2)N(C)C 10511,Cc1ccc(C#N)c(NC(N2CC(N3CCOCC3)C(O)C2)=O)c1 10512,N1(C(C(C)OCC=C)=O)CCN(C(c2sc(=N)[nH]c2C)=O)C(C(F)F)C1 10513,Cc1cc(C(=O)NCC=CCNC(c2c(C)[nH]c(C)c2C)=O)ncc1Br 10514,C1(NC(CC(C)(C)NC(CCN(C)CC)=O)=O)CCCCC1(C)O 10515,N1(C(C2CCC(C)(C)O2)=O)CCCC2CN(C(c3c[nH]nc3Br)=O)CCC12 10516,c1(C(N(CCOC)CCNC(C2CCC(OC)CC2)=O)=O)cc(C)nc(C)n1 10517,N1(C(c2cccc(NC(C)=O)c2)=O)CC2CC(NC(c3scnc3C)=O)C1C2 10518,CCCCC(C(=O)N1CCC(CCO)CC1)NC(c1cn(C)nc1OC)=O 10519,C1(C(N2CC3C(NC(c4ccc(=O)oc4)=O)C3C2)=O)COc2ccc(O)cc2O1 10520,Cn1cnc2[nH]c(=NCC3CCCN(C(=O)CSCC(F)(F)F)C3)nc(O)c12 10521,C(=O)(CCC(O)C(C)(C)C)N1CCC(C(C)NC(CN(C(COC)=O)C)=O)CC1 10522,N1(C(c2c(CNC(CC=CC=C)=O)ccs2)=O)CC2CCC(CO)(C2)C1 10523,c1(OC)ccc(COCC(O)CNC(C2(c3ccccc3)CC(C)C2)=O)cc1 10524,c1(C(=O)NCC(CO)NC(c2ccc(C(C)(C)C)nc2)=O)ccc(Cl)c(F)c1 10525,Cn1cc(C(C(=O)NC2CC(=O)NC2=O)N(C2CC(C(=O)OC)C2)C)c(I)n1 10526,CCCC(CN=c1cccc(S(=O)(=O)NC2CCc3ncsc3C2)[nH]1)OC 10527,C1(CC(=O)N(CCOCCNC(c2c(C)csc2)=O)C)CCCC(=O)N1 10528,CCC(CC(F)(F)F)N=c1[nH]c(=NC(C)CCc2ccccc2)[nH]c2c1CCC2 10529,C1(C(=O)NCCCOCCNC(C(C)C2=CCCC2)=O)CCC2(CC1)CC2(F)F 10530,C1(C(=O)Nc2ccc(-c3c(C)ncs3)cc2)CCCC12CCOCC2 10531,CC(C)CN=C(NCC1(Cc2cn(C)nc2C(F)(F)F)CCC1)NCC(C)(C)C 10532,CC(CO)C(=O)NCCOCCCN(C)C(c1cnn(C)c1)=O 10533,C=Cc1ccc(C(=O)NCC(C)(O)CNC(=O)COCCc2ccccc2)cc1 10534,C(CCCC(=O)NCCN(C(=O)CCS(C)=O)CCSC)N(C)C.N(C)C 10535,n1(CCC(=O)N(CC(C)NC(=O)C(Cl)=CCl)C)c(=O)nc(O)c2ccccc12 10536,c1(OC)c(F)cc(F)c(C(=O)Nc2c[nH]nc2C(N2CCN(C)C(C)C2)=O)c1F 10537,c1(C(N2CCC(OCc3ccccc3)C2)C(=O)NCC)cc(Cl)nn1C 10538,c1(CC)nocc1C(=O)N(C)CC1CCCC1NC(=O)CC1CNC(=O)O1 10539,c1(C(N(CC=C)CC=C)=O)ccc(Sc2ccc(C(F)(F)F)cc2)cc1 10540,c1(C(=O)NC2COCCN(C(C34CCCC3C4)=O)C2)ccc(=O)n2c1CCC2 10541,CN(N)C(=O)C(O)CC1CCN(C(=O)OC(C)(C)C)C1 10542,C1(C(=O)NC2(CCCC)CC2)CN(C(=O)C(C)OCCOC)CC1(C)C 10543,Cc1ccccc1C(=O)NC(CCN(C)C)C(=O)N1CC(C)C(F)C1 10544,c1(CNC(NCC2CC(CC)C2)=NCCF)nnc2c(=O)[nH]ccn12 10545,c1(C(N2CCCCC2COC)C(=O)NCCC)ccc(C)c(OC)n1 10546,CC1CN(C(C2CC23CC(C)(C)C3)=O)CCC1NC(C1CC2(CCCO2)C1)=O 10547,CC1CC=C(C(=O)NCC(C)(CO)NC(=O)CN2CSCC2=O)CC1 10548,c1(OC)nc(N(C2(C#N)CCNC2)Cc2c(F)cccc2F)ncc1F 10549,N1(C(c2nc(C)n(C)c2C)=O)CC2CCCC2(NC(C2CCCC(=O)N2)=O)C1 10550,N1(C(c2c(CNC(C(C(C)C)SCC)=O)nnn2C)=O)CC(C)C(C)(CO)C1 10551,c1(OC)ncc(NC(C2(F)CCN(C(c3cc(O)ncc3Br)=O)CC2)=O)cc1F 10552,C1(CC(=O)NC(c2cnc(C)s2)C)(NC(c2cocn2)=O)CCCCC1 10553,CC(=NO)C1CC(C(=O)NCC(C2CCN(C(=O)CNC=O)CC2)(C)C)C1(C)C 10554,c1(CC(N2CCN(C(c3n(C=C)nnc3)=O)CC2)=O)ccc(Br)c(O)c1 10555,N1(C(c2c(C)cc[nH]2)=O)CCC2(CC1)CC2CNC(c1cnc(S)[nH]1)=O 10556,c1(C(=O)NC2CC(C)CN(C(=O)C=Cc3cccs3)C2)cncc(P(C)(C)=O)c1 10557,N1(C(C(C)NC(CC)=O)=O)CCOCCC1C(=O)NCC1CC1c1ccccc1 10558,N1(C(C2CCCC(OC)C2)=O)CCCC(NC(c2cc(Cl)cnn2)=O)C1C 10559,c1(CNC=O)c[nH]nc1C.N1(C(=O)OC(C)(C)C)CCC1C(F)(F)F 10560,c1(C(=O)NCCC(C)NC(c2c(C3CC3)cccc2F)=O)cn2cccnc2n1 10561,C(=O)(C(O)CCS(C)=O)N(C1CCN(C(c2ncc(F)cc2N)=O)CC1)CC 10562,C(C(=O)NCCN(C(C1CCC12CCC2)=O)C(C)C)(C(F)(F)F)OC(C)=O 10563,C#CCC(O)C(=O)N1CC(C(=O)NCCCCC2CC2)C(F)C1 10564,N1(S(CCCC)(=O)=O)CCC(C(=O)NCCc2nccs2)(CO)CC1 10565,c1(CC)nccnc1C(=O)NC1CC12CC(NC(=O)C(C(C)C)C1CCC1)C2 10566,C1(C(=O)NCC2(CCNC(=O)C3=CCCSC3)CC2)CCc2ccccc2O1 10567,C1(C(=O)OC)CC(C(=O)NC(C)CCNC(C23COCC(C2)C3)=O)C1(C)C 10568,C1(C(=O)NC2CC(NC(=O)C(C)C(=O)N3CCOCC3)C2)(COC)CCCCO1 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10638,Cc1ccc(CNC(=O)C=CCC2(NC(=O)C(C)CC#N)CCC2)cn1 10639,c1(C(=O)NC(c2cccnc2)CN(C)C)c[nH]nc1C1CCOCC1 10640,N1(Cc2n(CC)nnn2)CC(OC)C(NC(C)=O)C1 10641,C1(NC(CCSCCC)=O)CCC(N(C)C(c2coc(O)n2)=O)C1 10642,C(=O)(CCCCCC1CC1)NCCC(CNC(C(c1cccc(C)c1)C)=O)O 10643,c1(C(C(=O)NC(CC(C)NC(C(Br)=C(C)C)=O)C)O)cccc(C)c1 10644,C1(C2CCN(C(C3CCC4(CC4)C3)=O)C2)(NC(c2cn(C)c(=O)cc2)=O)CC1 10645,c1(C(=O)NC(CNC(CCOCCOCC)=O)C)cc(C2CC2)no1.O(C)CC 10646,c1(C(N2CC(F)(CNC(C3CC(C)OC3)=O)C2)=O)cc2c(s1)CCC2=O 10647,c1(C(=O)NC2(CC(=O)NCCC34CC(CO3)C4)CCCC2)ccc(Cl)cc1O 10648,C1(C2CN(C(C34CCCC3C4)=O)C2)(NC(CCCn2c(C)ncc2)=O)CC1 10649,C(=O)(C(CC)CC(C)C)NCc1cc(C(=O)NC(CCC(=C)C)C)on1 10650,c1(C(=O)NCCN2CCN(C)CC2)nn2ccccc2c1NC(C1CC(O)CN1)=O 10651,C(=O)(CCN(CCO)C(c1cocn1)=O)NCCN(C)C 10652,C1(NC(CCC#C)=O)COC2(CCN(C(c3cncn3C(C)C)=O)C2)C1 10653,CCCCC(C)C(=O)N1CC(C(C)NC(=O)C(c2cnn(C)c2)O)C1 10654,Cc1ncnc(C(=O)NC(C)(C)CC(N2CCOC(C)CC2)=O)c1C 10655,c1(C(N2CCN(CCNC(C(CC)(C)CC)=O)CC2)=O)cnn2c1CN(C)CC2 10656,C1(C(N(CCNC(C(C)OCCC=C)=O)C2CC2)=O)CC=CC(O)C1 10657,c1(C(=O)NCC(CNC(C(C)=C(C)C)=O)O)oc(-c2ccccc2)nc1C 10658,Cc1nc(C)c(CCC(=O)NC2C3CC2N(C(=O)CC2CC(C)(C)C2)C3)c(O)n1 10659,C(=O)(CCC1=NNC(=O)CC1)N1CC(NC(C(CCCCC)O)=O)CC1(CC)CC 10660,N(C(=NCCN(S(C)(=O)=O)C)NCc1ccsc1C)Cc1cccc(C)c1 10661,c1(CC(C(=O)NCC(=C)CCNC(c2oncc2CC)=O)C)ccc(Cl)c(Cl)c1 10662,Cc1ccc(O)c(C(=O)N(C2CCCN(C(=O)CC#N)C2)CCO)c1 10663,c1(C(=O)NCC(CC=C)NC(c2c(C(F)F)cnn2C)=O)cc(C#N)ccc1Cl 10664,C1(C(=O)NC2CC(NC(c3cnc(SC)n3C)=O)C(O)C2)CCCCN1N=O 10665,c1(-c2nc(CCNC(=O)NCCCc3ccnc(C)n3)sc2)c(Cl)cccc1Cl 10666,CC1CN(C(c2cnc(OC3CC3)cn2)=O)CCN1C(=O)CS(N)(=O)=O 10667,C1(NC(C2(CO)CCN(C(CCC#CC)=O)C2)=O)CC2(CC(OC)C2)C1 10668,S(=O)(=O)(c1ccc(NCC(C)N(C)C2CC2)cc1Br)N(C(CC)C)C 10669,N1(C(c2c(C(C)(C)C)n[nH]c2)=O)C2CCC1CC(NC(C1CC3(CCC3)C1)=O)C2 10670,n1(CC(=O)N(CCNC(=O)C(c2ccc(C)cc2)C)CC)cnc2ccccc12 10671,c1(C(N2CC(NC(c3ccc(C)cc3F)=O)C(C)C2)=O)ccc(Br)c2cc[nH]c12 10672,Cc1ccc(C)c(C(N2CC(F)(C(=O)NC(C)Cn3cc(C)cn3)C2)=O)c1 10673,C(=O)(C(CC)CC(C)C)NCCNC(c1cn(CC(OCC)OC)nc1)=O 10674,c1(C(N2CCC(NC(c3cnc(C(C)O)s3)=O)CC2)=O)ccc2ccccc2c1 10675,C1(C(N2CCCC2CNC(C23CC4CC(CC2C4)C3)=O)=O)CCOC2(CCC2)C1 10676,c1(C(=O)NC2CCN(C(C(N3CCSCC3)C)=O)C2)nnn2c1CCCC2 10677,c1(C(N2CC3CC3C3CC23)C(=O)NCCCOC)ccc2c(c1)COC2 10678,c1(C(=O)NC2CCCC2CNC(=O)C(=O)C(F)(F)F)cc(F)cc2ccoc12 10679,N1(C(C2C(OCC)C2)=O)C(CO)CSCC1c1ccccc1 10680,c1(C(N2C3CC(NC(CCCC)=O)C2CC3)=O)c(OC)cnc2ccccc12 10681,c1(CNC(C(C2(O)CCC2)NC(c2cccnc2S)=O)=O)ccc(CO)nc1 10682,C(=O)(CCCCC(=O)NC1CCN(C(=O)CN2CCN(C)C(=O)C2)CC1C)OC 10683,c12cccc(c1)CC(=O)NC1CCC(C1)CC1(CC1)C(=O)N2.CC(C)=COCC 10684,C1(C(=O)NC(CCC)(C)CO)CCC(C)(C)N(C(=O)Cc2ccoc2C)C1 10685,C12(NC(c3cc(C)c(C)o3)=O)COCCC1CN(C(=O)Cc1[nH]cnc1C)C2 10686,c1(C(N2CCC(Cc3ccccc3Br)C2)=O)ccnc2ncnn12 10687,C=CCC(C)(C)C(=O)N1CCN(C(=O)C(C2CCC2)OC)C(C2CC2)C1 10688,N1(C(CSCC)=O)CCC(CC)(NC(=O)CCCCCSC)CC1 10689,CCC(C)(C#N)C(=O)NC1CC2(NC(c3cccc(C4CC4)c3C)=O)COC1C2 10690,c1(CC(=O)NC(C)CC(C)NC(=O)CCCCCO)ccc2c(c1)COC2 10691,Cc1oc(C(=O)NC2C3CC2N(C(=O)CCCN(C)C)C3)cc1S(C)(=O)=O 10692,N1(C(C(c2ccccc2)C)=O)CCC2(C1)CN(C(C1(F)CCCOC1)=O)C2 10693,C1(C(NOCC#C)=O)CCC(CNC(=O)CCc2cccs2)C1 10694,N1(C(Cc2c(C)ccs2)=O)CCCC2CN(C(=O)C=Cc3ccccc3)CCC12 10695,C12(NC(C3N(C(C)=O)CCCC3)=O)CCN(C(c3ccc(CO)nc3)=O)CC1C2 10696,c1(C(=O)NCC2CCN(C(CC3(C(=O)OC)CC3)=O)C2)cc(C#N)ccc1O 10697,c1(CNC(C2CCCCS2)=O)ccccc1-n1cc(CN2CCCC2=O)nn1 10698,C1(n2cc(C(CCC)C)nn2)CON(C(=O)C(C)C(F)F)C1 10699,C1(C(N2CC(C(N(C)C)=O)C2)=O)CCN(C(=O)CCc2ccc(Cl)cc2)CC1O 10700,c1(C(N(C2CCN(Cc3scnc3Cl)C2)CC)=O)cc(-c2cccnc2)no1 10701,Cc1oc([N+](=O)[O-])cc1C(=O)N(C1CCN(C(C2CC(F)C(=O)N2)=O)C1)CCO 10702,N1(C(=O)CCc2nc[nH]n2)C2CCC1C(F)C(NC(C1(CCNC=O)CC1)=O)C2 10703,N1(C(Cn2cc(C(=O)OC)nn2)=O)CCCC2(CCN(C(=O)C(C)C3CC3)C2)C1 10704,C(=O)(N=c1[nH]c(Cl)ncc1O)C1N(C(c2c(OC)ccs2)=O)CC2(CC2)C1 10705,C(=O)(C(O)C(F)F)N(CCN(C(C)C)C(c1ccc(NC(C)C)nc1)=O)C 10706,c12cnc(cn1)c(=O)n2C1CC1.C1(OC)CC2C(OCc3ccccc3)CC12 10707,C1(=O)NN(C(=O)C(CC(C)C)c2c(C)nn[nH]2)C(=O)NCC1 10708,CCCCCC(O)C(=O)NCC1CCN(C(c2coc(C)n2)=O)CC1O 10709,C=CCCC(C(=O)N1CC(C)(C)C1COC)NC(C1(C)CCC2CC2C1)=O 10710,c1(C(=O)NCC(C)(C)NC(C2C(=C)CC2)=O)cc2ccc(Cl)cc2o1 10711,C1(NC(c2cc(C(F)F)ccn2)=O)CCN(C(C2C(Cl)(Cl)C23CC3)=O)CC1F 10712,c1(SC)nc(N(C)CC2CCN(C(c3cnc(C(N)=O)cn3)=O)CC2)ncc1C 10713,N1(C(c2c(C)cco2)=O)CCC2CC(CNC(C3(C(F)F)CCC3)=O)CCC2C1 10714,Cc1onc(C(=O)NCC2CCCC(NC(C3CC(C)(C)C3)=O)C2)c1[N+](=O)[O-] 10715,Cc1ccc(C)c(C(c2nnnn2CCC2CC2)NCCOC2CC2(F)F)n1 10716,CN1CCCC(C)(C(=O)N(C)CC2(O)CCN(C(=O)CCc3cncs3)C2)C1 10717,C(=O)(CCN=C(NCc1ccc(Cl)cc1)NCC1CCC(C)CO1)NC(C)C 10718,OCC(Cc1cccc(F)c1)CN=c1[nH]c2c(F)c(F)c(F)cc2s1 10719,c1(C(=O)NC2CC3CN(C(c4c(C(C)C)ocn4)=O)C2C3)nccn2ccnc12 10720,N1(C(C(Cn2cccn2)NC(CC2(C)CC2)=O)=O)CCCC(F)(F)CC1 10721,N(C(=NCCCCl)NCCCN1CCCC1=O)C(C1CCOCC1)C#C 10722,c1(OC)cc([N+](=O)[O-])ccc1CNC(=O)C=Cc1ccc(Cl)cc1F 10723,C(=O)(C(C)(C)CC#N)N1C(CN(C(=O)Cc2cnc[nH]2)C)COCC1 10724,C1(OC)(CNC(=O)CC2CCC2)CCN(C(=O)CC(N2CCCS2(=O)=O)C)C1 10725,CS(=O)c1ccccc1-c1cccc(NCc2cncc(-c3ccccc3)c2)n1 10726,c1(OC)ncccc1NC(c1cc(CCNC(C2CCC2C(C)(C)C)=O)on1)=O 10727,C1(N(C)C(=O)NCc2ccncc2)CCN2CCCCC12 10728,c1(OCC)cccc2ccc(NCc3cnn(-c4ccccc4)n3)cc12 10729,C=C1CC2(C1)CC(C(=O)NC1CCN(C(=O)C=Cc3cncs3)CC1C)C2 10730,C(=O)(C(C)(C)C1CCN(C(c2cnn(CC)c2)=O)C1)NC(c1ccccc1)CC 10731,C1(OC)CCN(CC(O)COc2ccc(-n3cccn3)c(C)c2)C(C)C1 10732,C1(C(=O)NCn2cc(CC)nn2)CN(C)CCN1C(=O)C=CC(C)(C)SC 10733,C1(O)(CCNC(C(CC)OCC)=O)CCN(C(c2cnccc2Br)=O)C1 10734,N1(C(C2CCN2C(C2(F)CCCC2)=O)=O)CCC(CN2CCCC2)CC1 10735,CC1CN(C(C2(O)CCSCC2)=O)CCC1CNC(=O)Cc1cnc[nH]1 10736,C(=O)(C1CCCc2ccnn21)N1CC(C2CN(C(CS(C)(=O)=O)=O)C2)C1 10737,Cc1nnc(CN(CC(N2CCCC(CNC(=O)CC3CCOC3)C2)=O)C)n1C 10738,C(=O)(C1=C(F)CN(C(C2CCCC(=O)C2)=O)CC1)N(C)Cc1cscn1 10739,C1(C(=O)NC(CCOC)(C)C)CC2CC1CN(C(c1ccncc1F)=O)C2 10740,C(=O)(CCCC(C)(C)C)NCC(CC=C)NC(=O)C(=Cc1ccco1)C 10741,C#Cc1cn(C)nc1C(=O)NC1CCC(CC(N2CCCC2C)=O)C1 10742,CC1(F)CCCCN(C(c2ccc(C(F)F)cc2)C(=O)NC2CCOCC2)C1 10743,C#CCCCCC(=O)NCC1(CNC(c2ccncc2C)=O)CC1(F)F 10744,N1(C(C2N(C(CC(=O)OC)=O)CCC2C)=O)CC2CSCC(C2)C1 10745,N1(C(C2C(CC)C2)=O)CCCC2(C1)CN(C(c1ccc(N)cc1F)=O)C2 10746,c1(N(CC(=O)NCC2C(NC(CSc3cn(C)nc3)=O)C2)C)ccnc(Cl)n1 10747,Cc1cnn(CCCNC(=O)C=CCN(C(=O)CCCC2CC2)C)c1 10748,CCC(C)CC(=O)NCC(c1ccc(C(=O)NOCC(F)(F)F)cc1)=O 10749,C(=O)(C(O)CCC(F)(F)F)N1CC(CNC(c2c(C)cccn2)=O)N(C)CC1 10750,CCC(CC(C)C)C(=O)N1CCC(F)(CNC(=O)CC2CC(SC)C2)CC1 10751,N1(C(CCOc2cc(C)on2)=O)CC2(CC(NC(=O)C3=CCCCO3)C2)C1 10752,CC1OCCC1(C)C(=O)NC1CCOC(C(=O)N(C)CCc2ccncc2)C1 10753,C(CCN=c1[nH]c(=NCCC(C)F)[nH]c2c1COCC2)N(C(C)=O)C 10754,CCCC(CC)C(=O)N1CC(NC(c2cc(Cl)cc(Cl)c2)=O)CC(F)C1 10755,c1(OCC)ccc2ccnc(C(C(=O)Nc3ccccc3)N(C3CCC3)C)c2c1 10756,c1(C(N2C(CNC(c3cc(CCC)on3)=O)C=CC2)=O)n[nH]c2c1COC2 10757,N1(C(C(C(C)C)F)=O)CCCN(C(=O)COC(C)(C)C)C(c2ccccc2)C1 10758,C(CC(C)C)(C(=O)N1CC2(C1)CN(C(=O)Cc1cscc1Br)C2)OC 10759,CCC(O)C(C)C(=O)N1CC(CNC(=O)CN2CCCC(OC(F)F)C2)(OC)C1 10760,C(=O)(C1=COCCO1)NCC(C(C)(C)C)NC(c1c(Cl)cncc1Cl)=O 10761,C1(CN(C(CCC=C)=O)C)CCN(C(=O)C(c2ccc(F)cc2)CO)CC1 10762,N1(C(C2(NC(=O)C(F)C3CCCC3)C(C)(C)C2)=O)C2CCC1COC2 10763,N1(C(c2c(C(C)(C)C)ocn2)=O)CC2CC(NC(c3cscn3)=O)C(C2)C1 10764,C12(C(=O)NCCC3OCCN(C(C(CCSC)O)=O)C3)CCC(CC1)C2(C)C 10765,Cc1ccc(C(=O)NC2CN(C(c3ccn(C4CC4)n3)=O)CC2C)cc1F 10766,C1(CC(=O)OC(C)(C)C)(NC2CC3CC3C2)CCOCC1 10767,N1(C(=O)OC(C)(C)C)CC2COCC(C1)C2NC(=O)CCCc1ccc(F)cc1 10768,C(CC(=O)NC(C)(C)C(F)(F)F)(C(F)F)NC(C(CC)SC)=O 10769,c1(C(N(CCC)CCNC(C2CC(C3CC3)=NO2)=O)=O)nc2ncccn2n1 10770,C1(NC(C(COC)CNC(C)=O)=O)CCc2nn[nH]c2C1.C1(=O)C(C)(C)CN1C 10771,C1(NC(=O)NCCS(=O)(=O)NC2CCCC2)CCCC1C1CCCC1 10772,c1(N2CC3C(CNC(C(C)Cc4ccco4)=O)C3C2)ncnc(Cl)c1Br 10773,C1(NC(C(F)=C(C)C)=O)CC2CCC1C1CN(C(=O)C=CC3CCCC3)CC21 10774,N1(C(CC2N(C(c3cc(C)c(C)nn3)=O)CC2)=O)CCCC(O)(C2CC2)C1 10775,C(c1ccc(C)cc1C)=CC(=O)NCC1N(C(C=C(C)C(C)C)=O)CC=C1 10776,N1(C(c2c(CC)nccn2)=O)CCCN(C(=O)C(O)CC(F)(F)F)C(C)C1 10777,c1(C(=O)NCC2C(C)CCN2C(c2nnsc2N)=O)ccc(OC(F)F)cc1F 10778,C#Cc1ccc(C(N2CCN(C(=O)NC(C)(C)C)C(C(=O)OC)C2)=O)cn1 10779,Cc1cc(=O)n(C)cc1NC(=O)C(N1CCC(S(=O)(=O)NCC2CC2)C1)=O 10780,C1(NC(c2ccn(CCCC)n2)=O)CC(O)CN(C(c2ccc(CF)cc2)=O)C1 10781,N1(C(CCOC)=O)C2CC=C(C(=O)NC(c3cc(C)on3)C)C1CC2 10782,c1(CCC(=O)NC(CC(C)C)CNC(c2sccc2F)=O)c(F)cccc1F 10783,C(C(CC(C)C)C(=O)NCC1COCC1NC(c1cc(CC2CC2)on1)=O)OC 10784,S(=O)(=O)(c1ccc(N2CCOC(C)(C(C)(C)C)C2)c(Cl)c1)N(C1CC1(C)C)CC 10785,S(=O)(=O)(c1cc(C)c(OC)o1)N1CC(C(CC)CC)C1 10786,C1(C(n2cc(C(C)(C)N(C)C)nn2)C)COCCN(C(=O)COCC(=O)O)C1 10787,c1(C(N2CC(NC(C3(SC)CC3)=O)C(F)C2)=O)ccc2nc(O)[nH]c2n1 10788,C(CCN=c1[nH]c2c(c(=NCCN3CCOCC3C)[nH]1)COC2)OCC(C)C 10789,c12noc(C)c1N(C)C(=O)N1CCC(C3CCCCN3C2=O)C1.C1(CC)CC1 10790,Cc1nc(C(=O)NCCC(C)NC(C2CC2C)=O)c2n1CCCC2 10791,N1(C(CCCOCC=C)=O)CCN(C(=O)C(O)CC)C(CC(=O)NCC)C1 10792,C1(N(C(=O)CCCc2cccc(Cl)n2)C)CN(C(=O)CC(F)(F)Cl)CC12CC2 10793,N1(C(C(CC=CC)NC(=O)CC2CCC(=O)N2C)=O)CCCC(O)(CC)C1 10794,c1(CN=C(NCC23CC(CF)(OC2)C3)NC2CCC2)ncc2ccccn12 10795,C1(CNC(CC(=C)Br)=O)CCCC2(CCN(C(=O)C(C)CN(C)C)CC2)O1 10796,CCCCC(O)C(=O)NC(C1CCN(CSC(c2ccccc2)C2CC2)CC1)=O 10797,N1(C(C(C)(C)NC(=O)NCC)=O)CCCC(CNC(=O)C(C)c2ccsc2)CC1 10798,c1(CC)c(C(N2CCC(NC(=O)CSCC(F)(F)F)C(F)C2)=O)cccc1F 10799,c1(C(N(CCCNC(CC(CC)C)=O)CCO)=O)ncnc2cc[nH]c12 10800,S(=O)(=O)(c1ccc(=NCCc2ccc(OCCO)nc2)[nH]c1)N(CC(=C)C)CC 10801,Cc1cnc(C(N2CCC(NC(C3CCC(C)O3)=O)C23CC3)=O)c(C)c1 10802,CC1=NNC(=O)C1CC(=O)NC(CNC(=O)C(C)N1CC(C)C1)C(C)(C)C 10803,c1(CC(=O)N(C)CC2CCN(C(c3c(CC)n[nH]c3)=O)C2)cccc2nonc12 10804,C(C1CN(C(c2cc(C)c(O)nn2)=O)CC1C(=O)NCCC(O)C1CCC1)=CC 10805,c1(C(=O)NC(CNC(C2(OC(C)=O)CC2)=O)CO)ccc(CNC(C)=O)cc1F 10806,c1(CC)noc(COCC(=O)NC(C)(C)CNC(=O)CN2CC(C)C2)n1 10807,C=CC1(CO)CCN(C(=O)CCC(CC)NC(c2ccc(N)c(F)n2)=O)CC1 10808,C=CC(C)(C)CC(=O)NC(C1CCN(C(=O)CCS(C)=O)C1)(C)C 10809,C1(C(=O)NCC(C)N(C(=O)C(=O)N(C)C)CCC)CCS(=O)(=O)C1(C)C 10810,c1(C(=O)NCCC(C)N(C(CN2C(C)CC2)=O)C)nn(C)cc1N 10811,C1(CC)CCN(C(=O)CC(C)(C)O)C1CNC(c1cc(C)ncn1)=O 10812,C1(CN(C)C(C2(O)CCSCC2)=O)CC(F)CN1C(c1ccc(CO)o1)=O 10813,c1(COC(c2ccc(OC3CCOCC3)cc2)=O)cc2c(s1)CCOC2 10814,C1(OC)CN(C(=NCCCCl)NCc2ccc(CSC)cc2)CC1O 10815,Cc1c(C(=O)NC2CC(NC(c3ncoc3C3CC3)=O)C2)n[nH]c1C1CC1 10816,c1(C(=O)NC(c2cccc(C)c2)CNC(C(C)(C)SC)=O)nc(Cl)ccc1N 10817,FC(F)C(F)(F)CCN=c1[nH]c(N2CCOCC2)nc(=NCCc2cnn[nH]2)[nH]1 10818,c1(N(CC(=O)NCC(Cn2cc(C(C)OC)nn2)(C)C)C)ccc(Cl)cc1C#N 10819,C1(CNC(Cn2c(C)ccn2)=O)CC2(CC2)CN1C(c1cnn(CCO)c1N)=O 10820,C1(C(C)C)C(NC(c2cnn(C)c2N(C)C)=O)CCN1C(c1cnn[nH]1)=O 10821,C(=O)(C1=CCCC1C)N1C(CO)CC(NC(c2n(CC)c(O)nc2)=O)C1 10822,C1(C(N(CCNC(=O)C(n2nccc2C)C)CC)=O)Cc2nccn2C1 10823,C(=O)(CC(C)CC(C)(C)C)N1CC(NC(c2c(C)ccc(C)c2)=O)C(F)C1 10824,c1(C(=O)NC2C(CC(=O)NC(C#CCC)(C)C)CCC2)c(F)cncc1F 10825,c1(N2CC3(C(C(=O)Nc4c(C)ccc(I)c4)C3)C2)ncnc2c(C)csc12 10826,S(=O)(=O)(c1ccc(Cl)cc1)CC(=O)NC(C)CCNC(=O)C(C)OC(C)(C)C 10827,C(=O)(CCN(OC)C(=O)c1coc2c1COC2)N1CC(COC)(OC)C1 10828,c1(C(C)C)nc(C(=O)NCC(F)(F)C(F)F)n(-c2cccc(Br)c2)n1 10829,c1(C(C)NCC2(CC(=O)OCC)CNC2)csc(CC)n1 10830,C1(C(=O)NC(C=C)COC)CC(NC(c2cn(C)nn2)=O)CCO1 10831,c1(CN2CCCC(C)(C(=O)NC3CNC(=O)C3)C2)ccc(F)c2ccoc12 10832,Cc1cccc(OCC(=O)Nc2ccccc2CNC(=O)CC(C)(C)C#N)c1C 10833,c1(OC)c(Cl)ccc(C(=O)NCCC2CCC(NC(=O)C(O)CN(C)C)C2)c1F 10834,c1(C(N(CCC(C)NC(c2cnoc2C2CC2)=O)C)=O)cc(F)cc2nn[nH]c12 10835,c1(C(=O)NCCC(C)NC(=O)C(F)(F)c2csc(Cl)c2)cn(C)nc1Cl 10836,Cc1c(C(=O)NC(C2(O)CN(C(=O)CC(=O)N(C)C)C2)C)cnn1C1CC1 10837,C1(C)(C(=O)NCC(n2cc(-c3ccc(COC)cc3)nn2)C)COC(=O)OC1 10838,CC(C)(C)C(=O)N1CCCC1C(=O)N(CCC=CBr)C1CC1 10839,C(CC(C(=O)NC(c1ncc(F)cn1)C)NC(c1ccoc1Cl)=O)=CC 10840,N1(C(C2NCC(OC)C2)=O)CCC(C2(O)COC2)CC1 10841,C1(C(=O)NC2C(NC(c3cc(OC)ns3)=O)C2)CN(Cc2ccccc2)CCN1 10842,C1(CNC(CCCOC(C)C)=O)CC(C)(C)CN1C(=O)CC1(O)CCCOC1 10843,C1(C(C)C)CN(C(C2CC2(C)C(F)F)=O)CC1C(=O)N(C)Cc1cnn[nH]1 10844,N1(C(c2scc(C)c2)=O)CCC(NC(c2cnc(C3CC3)s2)=O)CC1C1CC1 10845,C1(NC(CC=CCC)=O)CC(O)CN(C(=O)C(=O)Nc2ccccc2)C1 10846,N(C1CCSc2ccc(F)cc21)C(C(=O)Nc1cc(C(F)F)c(Cl)cn1)=O 10847,c1(C(=O)OCC)ccc(C(=O)NC2CCC(CC)(NC3(CO)CC3)CC2)c(O)c1 10848,CCCCC(C)CCC(=O)N(C1CC(C(=O)NCC(CC)SC)C1)C 10849,c1(NC(=O)NCC2CC2c2ccc(Cl)cc2)cc([N+](=O)[O-])sn1 10850,CC1CC2(CC(C(=O)NCC3(C)CCN(C(=O)CCC4CC4)C3)C2)C1 10851,CC1CCN(C(c2cc(Cl)cs2)=O)CCN1C(=O)CC1OCCCC1(C)C 10852,C1(CNC(c2c(C)n[nH]c2C)=O)CN(C(c2ccnc(C)c2N)=O)CC12CC2 10853,CC(C)(CCC#N)C(=O)NCCOCCNC(=O)CC1CCC2CC12 10854,Cc1ccc(S)cc1.C12(C=O)CCC1CC2.n12cc(nn1)C1CC(C1)NC(=O)C2 10855,N#Cc1ccc(COCC(=O)OCCCOc2ncc[nH]2)cc1 10856,C1(NC(C=CS(CC)(=O)=O)=O)CCC2CCN(C(=O)C(=Cc3cnc[nH]3)C)C1C2 10857,C1(N(CCC)C(c2cc(C)co2)=O)CCN(C(=O)CSCC2CCCCO2)CC1 10858,C1(C(N2CC(C(C)OC)C2)=O)CC(C)(C)CCN1C(c1cccc(C)n1)=O 10859,Nc1c(C(=O)NC2CC(CCNC(=O)CN3CCCC3CO)C2)cc(F)cc1Cl 10860,c1(CC(C(=O)C(C(N2CCSCC2)C)=O)O)ccc(F)cc1.C1(N)CC(N)C1 10861,c1(NC(=O)Cc2cc(F)cc(Br)c2)ccc(OCC(F)F)cc1F 10862,c1(OC)cc(C)cc(C(=O)NCC=CCNC(c2cnc(C)nc2CO)=O)c1N 10863,C(=O)(C(C)(C)C(F)(F)F)NC1CN(C(c2nc(CCC)oc2)=O)C(C)C1 10864,Cc1cc(C(=O)NC(C)(CNC(C2CC2C(N)=O)=O)C(C)C)cc(C)c1C 10865,Cc1cc(C(=O)NCC2(CNC(=O)CC3COC(=O)C3)CCC2)n(CC(F)F)n1 10866,N1(C(C(CC)=CC)=O)CCC(C)C(NC(c2cc(Cl)cc(Cl)n2)=O)C1 10867,C1(CC(=O)OC)CC(C)(C)CN1C(=O)NC(C1(n2cccn2)CC1)C1CC1 10868,C1(NC(CCNC(N)=O)=O)CCCCC1NC(C1(CO)CC(F)(F)C1)=O 10869,C(=O)(C(=O)N1OC2CCC1C2)NC(C(C)C)Cc1ccc(F)cc1 10870,C1(N(C)C(c2ncoc2C2CC2)=O)CCCC(NC(=O)C=Cc2cncn2C)C1 10871,c1(C(N(C2CCN(C(=O)CC3CC(CF)C3)CC2)C)=O)nncc2c1CCCC2 10872,C1(NC(Cn2c(C)cc(C)n2)=O)CC2CC1CN(C(c1cnsn1)=O)C2 10873,C1(C(=O)OC)CCC2(CCC2)N(C(=O)CCC2CCOC2=O)C1 10874,CC1CN(C(c2csc(-c3ccc(Cl)cc3)n2)=O)CC(C)N(C(=O)CNC=O)C1 10875,C1(NC(C2(C)CC(NC(C(C(C)C)O)=O)C2)=O)CC(C)CCC1O 10876,c1(CC)nc(N2CCC(NC(C3(C(N)=O)CC3)=O)C(C)(C)C2)c2ccsc2n1 10877,C(=O)(CS(=O)C(F)(F)F)N1CCC(CNC(CCOC)=O)C1(C)C 10878,Cc1cc(OCC(=O)NC2CC(NC(C3CCOC(=O)CC3)=O)C2)ccc1Cl 10879,C(=O)(CCC[N+](=O)[O-])N1CCC(C)(CNC(C(Cc2c(C)noc2C)C)=O)C1 10880,C1(CC(=O)NC(C(=O)NCC(C)C)c2cn[nH]c2)CC2C=CC1C2 10881,Cc1nn(C)c2c(N3CCOc4ncccc4C3)nc(=NCc3cc[nH]n3)[nH]c12 10882,C(N=c1[nH]c(N(C)CCNC(=O)C2CC2)nc2cc[nH]c12)c1cc(C)c(CO)cc1 10883,c1(CN=[N+]=[N-])ccc2c(c1)CCO2.C(=O)C(C)(O)C(F)(F)F.CC(C)C1CC(=O)N1 10884,C1(CNC(COCCOCC)=O)CC2(CCN(C(c3cnc(Cl)s3)=O)C2)CO1 10885,C1(n2cc(CNC(C(C)=C(C)C)=O)nn2)CCN(C(=O)CCc2cccs2)CC1 10886,C1(CNC(C2(OCC)CCCC2)=O)CN(C(c2c(C(C)C)n[nH]c2C)=O)CC1C 10887,c1(CC(N2C(CNC(C(C(C)C)(C)O)=O)COCC2)=O)cccc2c1OCCO2 10888,N1(C(CN(C(C)=O)C)=O)CCC(C2N(C(=O)CC3CC3(C)C)CC2(C)C)CC1 10889,N1(C(C(c2c(C)n[nH]c2C)C)=O)CCCN(C(c2cnns2)=O)C(C)C1 10890,C1(C(N2CC(CNC(=O)CSC)C(C(F)(F)F)C2)=O)(COC)CC=CCC1 10891,c1(OC)cc(CCC(=O)NC(C)C(CO)NC(c2nncs2)=O)on1 10892,Cc1ccsc1C=CC(N1CCC(OCCNC(=O)CC2CCCO2)C1)=O 10893,C12(OC)CC(C1)N(C(N1CCC(C(=O)NON3CCSCC3)(C(C)(C)C)C1)=O)C2 10894,CCC(C)CCC(=O)NCC1COCCN1C(c1cnc(-c2ccccc2)[nH]1)=O 10895,C1(C)(CNC(C(=O)NC(C)C)=O)CCC(NC(=O)C(c2ccccc2)=O)C1 10896,c1(CC(=O)NCCCCNC(c2ccc(C#C)cn2)=O)cn2cc(C)sc2n1 10897,C1(CNC(CCNC(CSCCOC)=O)=O)CCN(C(N)=O)C1 10898,Cc1cccc(CCN(CCCNC(c2ccc(C3CCCCC3)cc2)=O)C)c1 10899,C(CCCCC(=O)NCCc1cnc(C)s1)NC(C1(OC)CCC1)=O 10900,N1(C(C(C(C)C)F)=O)CC2CCCC(Nc3cc(-n4ccnc4)ncn3)C2C1 10901,CC(C)CC(C(=O)NC(C)CCc1cn[nH]c1)ONC(=O)COCC(C)C 10902,c1(CN2CC(C(N(CC)Cc3ccncc3)=O)SCC2)cnc(Cl)c(Cl)c1 10903,CCC(F)(F)CC(=O)N1C2CCC(C2)C1CNC(=O)C(C)Oc1ccccc1 10904,C1(C(N2CCC(NC(c3n(C)nnc3)=O)(CO)C2)=O)CCc2nccn2CC1 10905,c1(C(=O)NCC(C2CCC2)NC(C=C(CC)CC)=O)cc(F)ccc1Br 10906,c1(SC(C(=O)NCC2CC(NC(C(c3cnccn3)C)=O)C2)C)ccccn1 10907,C1(O)(C(N2C(C(N3CCCCC3CO)=O)CC2)=O)CCOCC1 10908,c1(OCC)ncccc1NC(C1CC(O)(CNC(=O)CN(C)CC)C1)=O 10909,Cc1ccc(C(=O)NCCOC(C)(C)CNC(c2nccnc2C)=O)c(Cl)c1 10910,c1(C(=O)NCCCN(CCO)C(C2CCCSC2)=O)ccc2nn[nH]c2n1 10911,N1(C(CC(C)F)=O)CCC(C)(C)CC1C(=O)NCc1cncc(C#N)c1 10912,C(c1ccccc1Cl)=C(C)C(=O)NC1CC(C)N(C(=O)CCn2ccc(=N)[nH]2)C1 10913,c1(C2(C(=O)NC3C=CC(CNC(=O)Cn4nccn4)C3)CC2)cc(F)cc(Cl)c1 10914,S(=O)(=O)(c1cccc(N2CCC3(CC2)CC3)n1)NCC1CCC(C)C1 10915,C1(C)(CC)CC(NC(=O)NC(C2(CC(=O)OC)CCOCC2)C)CCO1 10916,C12CCN(CC1)C2=O.C1(NC(COCc2nnc(C)s2)=O)CC12CC(O)C2 10917,c1(CN(CCC#C)C(c2cc(OC)ccn2)=O)cnc(N2CCCC2CO)c(Cl)c1 10918,CCC(C)C(CC(=O)N1CC(S(C)(=N)=O)C1)NC(C1CCC1C)=O 10919,C(=O)(CCCCC(=O)N1CC(CNC(=O)CN2CCCCC2)CC1C)OC 10920,c1(C(=O)NCC(CCC)NC(=O)CCN(C)CCC)c(C)coc1CC 10921,c1(CN(CCOC)C(=O)NCc2cncs2)ccc(F)cc1Br 10922,CC(C)C(C(=O)NCCC(C)NC(C1CCC(=O)C1)=O)NC=O 10923,N(C1COc2ccc(Cl)cc21)C1(c2n(CCSC)nnn2)CCN(OC)CC1 10924,c1(N2CCC(NC(C3CCC(OCC)CC3)=O)C2C)nc(C)nc2n[nH]cc12 10925,c1(C(N2C(CC)CN(C(c3cc(Cl)n(C)n3)=O)CC2)=O)cccc2ccncc12 10926,c1(CN2CC3C(C(=O)Nc4nc(O)cs4)C3C2)cccc(I)c1F 10927,C1(C(=O)NCC2CN(C(CN3CCC(=O)NC3=O)=O)C2)CNC(=O)CC12CCC2 10928,N1(C(c2cn(C)nn2)=O)CCCC(CNC(=O)CCC2CCC2)CC1 10929,c1(OC)ccc(C(=O)O)cc1CN1CCC(O)C(C(=O)Nc2nc(C)co2)C1 10930,C12(CNC(c3n(COC)ncc3)=O)CC1CN(C(C1CC(C)(O)C1)=O)C2 10931,c1(NC(c2cc(-c3c(OCC)cc(F)cc3)ncc2)=O)cc(Br)cc2[nH]ccc12 10932,Cc1nc2ccc(C(=O)NC3CN(S(=O)(=O)c4cccs4)C3)cc2o1 10933,CCC(C)(COC)C(=O)NC1CC2CC1N(C(c1ccc(C(C)(F)F)cc1)=O)C2 10934,N1(C(c2cncc(NCC)c2)=O)CCC(NC(C2(CCCF)CC2)=O)C(CO)C1 10935,C1(NC(C(CN(C)C)O)=O)(CO)CCN(C(=O)COc2ccc(F)cc2)C1 10936,c1(SCC)ncc(NC(=O)C=CCNC(=O)C(CN(C)C)N(C)C)cn1 10937,N1(C(c2c(C)nccc2Cl)=O)CCCC(NC(=O)C=Cc2ccsc2)C(F)C1 10938,N1(C(C(C)C2CCCC2)=O)CCC2CCC(C1)N2C(c1cc(=O)cc[nH]1)=O 10939,c1(C(C(=O)NCCN(CCC(=O)O)CC)OCC)cc(F)cc(F)c1 10940,N1(C(CC(=O)NCC#C)=O)CCC(C(=O)NCCCC(C)(C)O)C12CCC2 10941,N1(C(CC(C=C)C)=O)CC(C)N(C(=O)C2=NOCC2)CC1C 10942,N1(C(C2C(C)OC(C)C2C)=O)CC2CCC1C1CN(C(c3cc(Br)co3)=O)CC21 10943,c1(OC)ccc(CC(C)CN(C)C(=O)NCc2ocnc2C)cc1 10944,c1(CC(CN(C)C)=O)ccc(CCCC2C(C)C2)cc1 10945,CCCCC(F)C(=O)NC1CCCCC1C(N1CCC(CN=[N+]=[N-])C1)=O 10946,c1(CC(=O)NC2CCN(C(c3cscn3)=O)C2)noc2ccc(Br)cc12 10947,c1(OC)ccc(CN=C(NCc2ccco2)NCC2CC2C)cc1 10948,Cc1cc(C(=O)NC2CC3CN(C(=O)C(CO)C(C)C)CC23)cc2nn[nH]c12 10949,CCCC(C(=O)NC(C)CCNC(c1nn(CC)nc1Br)=O)NC(N)=O 10950,CN(C)S(=O)(=O)N1CCCC1CNC(=NCC1CC1)NCC1CCCN1C1CC1 10951,C(=O)(C(O)C1=CCCCC1)NC(C(=O)NCc1c(C)cnn1C)CC1CCCC1 10952,c1(C(=O)NCC2C(NC(c3cccc(O)n3)=O)C2)cc(Br)ccc1[N+](=O)[O-] 10953,c1(C(N2CCC(O)(CNC(Cc3scc(C)n3)=O)C2)=O)ccc(C(N)=O)c(Cl)c1 10954,c1(C(=O)NC(C(C(C)C)C)CNC(c2ccn(C)n2)=O)cc2ccc(O)cc2[nH]1 10955,C1(CCNC(c2ccn(C)n2)=O)CN(C(c2cccc(Cl)c2F)=O)CCCO1 10956,c1(C(N2C(C3CCN(C(C(C)NC=O)=O)C3)CCC2)=O)cccc(=O)n1C 10957,n1(CCC)c(C(N2CCC(CF)(NC(=O)C3=CCOC3)C2)=O)cc2ccccc12 10958,C(=O)(CCCn1cc(NCC(O)CNC(C)=O)cn1)OCC 10959,C1(CN(C(C2(Cc3ccc(Cl)cc3)CC2)=O)CC)CCN(C(=O)C(O)CF)CC1 10960,C(=O)(CC=CC(C)(C)C)NCC=CCNC(CC1(C)CC1)=O 10961,c1(C(N2C(C3(O)CN(C(c4ccn(CCC)n4)=O)C3)CCC2)=O)ccc(=N)[nH]n1 10962,C(N=c1[nH]c(=NCC2CCCSCC2)[nH]c2c1CC(C)CC2)c1[nH]c(=NC)sc1 10963,C1(N(C(CCN(C(C(COC)O)=O)C2CC2)=O)C)CCCC(C)C1C 10964,N1(C(CCOCC#C)=O)CC2CCC1CN2C(C1CCCC(C)CC1)=O 10965,S(=O)(=O)(c1ccc(NCCOc2cccc(Cl)c2)cc1Cl)NC(CCSCC)C 10966,C(=O)(CCCCC(N)=O)N1CCC(NC(c2c(C)ccc(OC)c2)=O)(CF)C1 10967,C(=O)(CCCC(C)(F)F)N1CC(N(C(=O)C=Cc2ccnn2C)C)C(C)(C)C1 10968,c1(C(=O)NC(C)CCNC(=O)C=CC2CC2)c[nH]c2cccc(Br)c12 10969,c1(C(N2CC3CN(c4nccnc4F)CC3C2)=O)c(F)c(F)cc(F)c1F 10970,C(=O)(CP(C)(C)=O)NC1(CCNC(CCc2n(C)ncc2)=O)CCCC1 10971,c1(N(C(C#C)C)C)nnc(-c2ccc(C)nc2)n1CC(=O)NCCO 10972,c1(C(=O)NCCC2(C)CCN(C(c3nocc3Cl)=O)C2)cc2c(s1)CCC2 10973,N1(C(C2(COC)CC(=C)C2)=O)CC=C(C(=O)N2CCC(CC)C2)C1 10974,c1(C(=O)OC)c(N2CC(CO)(NC(=O)C(c3ccccc3C)C)C2)ncnc1Cl 10975,C1(NC(C(CCCC)O)=O)Cc2ccccc2C1NC(C1(CC)CC1)=O 10976,C1(O)(CN(C(C(C)=C2CCCC2)=O)C)CCCN(C(C2CN(C3CC3)C2)=O)C1 10977,C1(C)(C(=O)NCC(C(C)C)NC(=O)C(C)S(N)(=O)=O)CC2(CCC2)C1 10978,N1(C(C(N)=O)=O)CCC2(CC1)COC(CNC(=O)COCC1CCCCO1)C2 10979,c1(CCNC(=O)NC(CO)CF)nc(-c2cccnc2)no1 10980,N1(CC(=O)Nc2n(C)nc(C(F)(F)F)c2)CCC(NC(c2ccsn2)=O)C(O)C1 10981,c1(C(N(C(C)CNC(c2cccc(O)c2)=O)C)=O)cccc2nsnc12 10982,C(=O)(C1Cc2ccccc21)NC(CCC=C)C(=O)NC1(C)CS(=O)(=O)C1 10983,Cc1ccc(SC(C)C(=O)NC2C=CCN(C(C3CCC(=O)NC3)=O)C2)cc1 10984,N1(C(CCC(=O)NCC(CNC(CC(C)C2CC2)=O)O)=O)CCc2sccc2C1 10985,c1(COC)nc(C)c(C(=O)NCCC(C(C)C)NC(c2n[nH]cc2C(C)C)=O)s1 10986,C1(NC(c2c(OC)n[nH]c2)=O)C2CCC1N(C(=O)Cn1ccc(Br)cc1=O)C2 10987,c1(C(=O)NC2CCN(C(C3CC3F)=O)C2)c(F)cc(C(F)(F)F)cc1Br 10988,n1(CC)cc(C2OCCC2C(=O)NC2CCCC2NC(=O)CN2CC(C)C2)cn1 10989,C1(C(=O)NC2(C)CC(NC(c3cc(Cl)ccc3Cl)=O)C2)CCC2(CCC2)O1 10990,c1(C(=O)NC(CNC(C2N(CC)CCCC2)=O)CO)nccc(OC)c1O 10991,S(=O)(=O)(c1ccc(NCCOc2ccccc2)c(C#N)c1)NCCSCC=C 10992,N1(C(C(C)(C)NC(=O)NCCC)=O)CCC(CNC(C23CC(F)(C2)C3)=O)C(C)C1 10993,c1(CCC(=O)N(C2CCC(NC(c3ncoc3C3CC3)=O)C2)C)ccc(F)nc1 10994,O=C(C#CC1CCCO1)N1CC2(CCN(C(C3(C(F)(F)F)CC=CCO3)=O)C2)C1 10995,Cc1noc(C)c1S(=O)(=O)N1CCOC2CN(c3ncc4ccsc4n3)CC12 10996,c1(C(=O)OCC(=O)N=c2cccn[nH]2)cc2c(nc1O)CCCC2=O 10997,c1(C(=O)NC(CC)Cn2cncn2)c[nH]nc1CCNC(C1(C)CC1)=O 10998,c1(CNC2C(C(N3CCC(Br)CC3)=O)CCC2)c(F)ccc(Cl)c1F 10999,C#CC1CN(C(=O)C(CNC(=O)CC2CCC(C)(C)C2)CC(C)C)CCN1C 11000,C(c1ccccc1Cl)=C(C)C(=O)NCC1(CNC(=O)CCCCN(C)C)CC1 11001,c1(CC(N2CC(CNC(C=CC=CC)=O)OCC2)=O)ccc(C)c(OC)c1 11002,C(C)(C)(CCC(=O)NC1CC2CC1CC2CO)NC(C1=CC(C)C1)=O 11003,c1(C(N2C3C(NC(c4occc4F)=O)CC(C3)C2)=O)cccc2occc12 11004,C(=O)(CCCCCN=[N+]=[N-])N1CC(C)N(C(C2(CCC)CC2)=O)C(C)C1 11005,C1(CNC(CC2N(C(C3CC(C(C)C)C3)=O)CC2)=O)CNC(=O)CO1 11006,c1(C(=O)NCC2C(C)CN(C(=O)CC34CCCC3C4)C2)ccc(Cl)c(Br)c1 11007,C1(C(=O)NCCOCCNC(c2cnc(CC)s2)=O)C(C2CC2)C1(F)F 11008,c1(C(=O)NC(CC(C)NC(C(C)=C2CCCC2)=O)C)c(C)nc(C(C)C)nc1S 11009,N1(C(C=CC=CCCCCC)=O)CCC2CCC(C1)N2C(=O)COCCCF 11010,C1(O)(CCC)CCN(C(C2CCCN(C(C3OCCCC3(C)C)=O)CC2)=O)CC1 11011,Cc1nccnc1-c1cn(-c2csc(-c3sccc3CO)n2)nn1 11012,Cc1nnc2n1CC(C(N1CCC(CCNC(C3CCCN3C3CC3)=O)C1)=O)C2 11013,N1(C(c2cnc(CC)[nH]2)=O)CC(C(F)F)CC1CNC(=O)CCCNCC 11014,C(=O)(C(C)C(C)(C)C)NC1C(NC(Cn2c(C(C)C)nnn2)=O)CC1 11015,N1(C(c2ccc(SC)cc2)=O)CCC2(CC1)CC2NC(=O)C(C)NC=O 11016,c1(C(=O)NCC2CC2CNC(c2cnc[nH]2)=O)cccc(Cl)c1 11017,C(C)(C(=O)OC(C)(C)C)(C(=O)NC1CN(C(C2CC3CC3CC2C)=O)C1)OC 11018,c1(C(=O)NC(CC)CN(C(=O)Cc2ccc(Cl)nc2)C)cnn2c1NCC(C)C2 11019,c1(C(C(=O)NC2CCN(CC(=O)NC)CC2)NC(CCC#C)=O)c(C)cccc1Br 11020,C1(NC(C(CN(CC)CC)F)=O)CC12CC(NC(C1(C)C=CCCC1)=O)C2 11021,c1(C(N(CCCCCC)CCNC(=O)C(C2CC2)C2CC2)=O)n[nH]c(C)c1Cl 11022,N1(C(C(C)Oc2ccccc2)=O)CCC(CNC(C2CC2C2CC2C)=O)C12CC2 11023,C=CC(C)(C)CC(=O)N(C(CC(F)F)C(=O)N1CCC(OC2CCC2)C1)C 11024,c1(C(N2CC(C)(CCC(=O)NC3CN(CCC)C3)C2)=O)cc2ccccn2n1 11025,N1(C(c2nc(C(C)=O)sc2)=O)CCC(C2CCN(C(=O)COCCO)C2)CC1 11026,c1(C(N2C(C)CCC(NC(c3c(C)coc3)=O)C2)=O)ccc2ocnc2c1 11027,c1(CC)ccc(C(=O)NC2CC23CC(NC(C2CC2C(N)=O)=O)C3)cc1CC 11028,N#Cc1cc2c(n(CNCc3nc4ccccc4n3C(F)F)c1=O)CCC2 11029,C1(NC(CC(=O)OC)=O)C2CCCC1CC(NC(C1CN3CCN1CC3C)=O)C2 11030,N1(C(C2CCN(C(CCC)=O)CC2)=O)CCN(C(C2CNC(=O)C2)=O)C2CCC12 11031,C1(n2cc(-c3cn(CC)nc3)nn2)CCCN(C(C2CCC(=O)CC2)=O)C1 11032,c1(NC(C2N(Cc3c(C)noc3)CCC2)=O)cc(Br)ncc1F 11033,C1(c2n(CC)nnn2)(NC(C2CCCC(C)O2)=O)CCN(c2cccc(C)n2)CC1 11034,c1(C(N2CCC(CCNC(C3(COC)COC3)=O)C2)=O)ccc(C(C)C)nc1O 11035,C1(C(=O)NC2C(NC(c3cccc(C(F)F)c3)=O)COC2)CS(=O)(=O)CC12CC2 11036,C1(NC(C2C(C)(C)CO2)=O)CC2(CCCCN2C(c2nnn(C(C)(C)C)n2)=O)C1 11037,Cc1c[nH]cc(C(N2CC(NC(=O)CSc3cn[nH]c3)CC(O)C2)=O)c1=O 11038,C1(C(=O)NC(C=C)CO)(CC)CCN(C(=O)CC2CCCCN2C)C1 11039,c1(CC)onc(C)c1C(=O)NC1CCN(C(=O)Cn2c(C)nccc2=O)C1C 11040,CC1(NC(=O)CCc2nccs2)CCN(C(=O)C(F)CC2CCCC2)C1 11041,C#CC1(NC(=O)C(C)(C2CC2)N(C)C(C2CC3CC3C2)=O)CCCCCC1 11042,c1(CC)cnoc1C(=O)NCCN(C(c1cc(C(C)(F)F)n[nH]1)=O)CC 11043,c1(CC(=O)NCC(O)CNC(c2csc(-c3ccoc3)n2)=O)ccc(F)cc1 11044,CC1(O)CCC(CC(=O)NCCNC(c2n[nH]c(C3CC3)c2Cl)=O)CC1 11045,c1(OC)cccc(S(=O)(=O)N2CCC3C2CCCN3C(=O)C(Cl)(Cl)Cl)c1 11046,N(C1CCc2c(C(=O)O)ccnc21)C(c1nc(-c2ccc(OC)cc2)sc1)=O 11047,c1(CN(C)C)cc(C(=O)NC2CCC(CNC(=O)C(F)CC3CC3)CC2)ccn1 11048,C(CCCC(=O)N1CCCC1C(N)=O)NC1CCCN(c2n(CC)nnn2)C1 11049,C1(CNC(c2ccc(CSC)cc2)=O)CC(F)(F)CN1C(=O)C(C)S(N)(=O)=O 11050,C1(C(=O)NCC2CC3CCC(C2)S3)C2CCCCCCC12 11051,Cc1cccc(Cl)c1C(=O)NC1CC(NC(=O)CCC2CCCCC2)C(O)C1 11052,C1(C(N2CCC(C)(O)CC2)=O)CC2(CCC2)CN1C(=O)CSCC(F)F 11053,C1(N(C(c2cccn2CC)=O)CC)CCCN(C(C2CCC2(F)F)=O)CC1 11054,C1(C(=O)NC2(C)CCCN(C(c3ccc(N)c(N)n3)=O)C2)CCC(C2CC2)CC1 11055,C1(CC)CN(C(=O)CN(C(=O)CCc2csnn2)C)CC1F 11056,CN1CC=C(CC(=O)N2CCCCC(N(C)C(C3COCCN3C=O)=O)C2)CC1 11057,C12(c3onc(C)n3)CCC(CC1)N2C(=O)C(c1cccc(O)c1)C 11058,c1(OCC)cnc(C(=O)N(C)CC2CCN(C(c3ccn(C(C)C)n3)=O)C2)cn1 11059,c1(C(=O)NCC2(F)CCCN(S(CC)(=O)=O)C2)cnc2[nH]c(C)nc2c1 11060,C1(C(=O)NC2(CN(CC)CC)CC2)COCCN(C(=O)C=Cc2ccnn2C)C1 11061,c1(C(N2C(CCS(C)(=O)=O)CCCC2)=O)ccc2c(c1)C(=O)OC2(C)C 11062,O=C1CCc2cc(C(N3CC(N4CCCC4=O)C3)=O)c(F)cc2N1 11063,c1(OCCC(COC)OC)nc2ccccc2nc1N1CCCC(F)(CO)C1 11064,c1(CNC(C(=Cc2ccco2)C)=O)ncccc1C(N1CCCC2CC12)=O 11065,C1(C(N(CC(=C)C)CC)=O)CC=CCN1C(=O)Cc1csc(C)c1 11066,C12(NC(CCc3n(C)c(S)nn3)=O)CCC(CN(C(c3ccc(F)s3)=O)C1)C2 11067,c1(N2CCC(N(CCC)C(c3ccnc(F)c3Cl)=O)CC2)nc(C)ncc1F 11068,Cc1cc(C(=O)NCC(C2CCCC2)NC(c2ccccc2F)=O)c(O)nn1 11069,CC(C)C(C)(CNC(C1CCCC(C)O1)=O)NC(=O)CO 11070,C1(C)(CNC(C2CCC(CC)O2)=O)CCCN1C(=O)CCc1ccccc1Cl 11071,C1(CNC(C(CC=CCC)C)=O)CC2CCCCC2N1C(=O)CCC(=O)C1CC1 11072,C1(CCC(N2CCC(CNC(C3CC(C)(C(=O)OC)C3)=O)C2)=O)CC(C)(C)CO1 11073,c1(C(=O)NC(C#C)CC2CCOC2)ccc(-c2ccc(Br)cc2)n1C 11074,C(=O)(C1=NOC2(CCC2)C1)NC(CC(C)NC(c1ccc(CC)c(OC)c1)=O)C 11075,C(c1ccc(Cl)cc1)=CC(=O)NCC1CC(OC)CN1C(=O)CCc1cnoc1 11076,Cc1nc(CC(N2CCC(C(=O)NCCC3CCCOC3)C2)=O)cs1 11077,Cc1cc(Cl)c(Cl)cc1C(=O)NC1CCCCC1NC(=O)CC1(C)CC1 11078,S(=O)(=O)(c1cccnc1NC1CCSC1)N1CCC(c2ccc(C(C)C)cc2)C1 11079,N1(CC=C(C)Cl)CC=CC1CF 11080,c1(OC)cc(C(=O)NC2(C)CCN(C(=O)C(C)NC=O)C2)cnc1O 11081,c1(C(=O)CNC(c2cccs2)=O)cc(Cl)ccc1OCC1CCCO1 11082,C1(C)(NC(C(CCN(C)C)NC(c2coc(CO)c2)=O)=O)CC2CCC1C2 11083,c1(C(N2C(C(N(C)CC3(C#N)CC3)=O)CCCC2)=O)ncc(C)cc1C 11084,C(=O)(CCCN(C)N=O)N1CCC(C)C1CNC(c1cnn(-c2nccs2)c1)=O 11085,N1(C(C(CC)=CCCC)=O)CCC(N=[N+]=[N-])(C(N2CCC(CC3CC3)C2)=O)C1 11086,N(C1CCOc2cc(F)cc(F)c21)C(=O)NCC#CCCCCCC 11087,N1(C(c2c(C)[nH]nc2I)=O)CCOC2(CCN(C(=O)C(N)=O)C2)C1 11088,N1(C(C(C#N)CC2CC2)=O)CCN(C(=O)Cc2cccc(F)c2)CC1C1CC1 11089,C#CCC(C)(C(=O)N1CCN(CC)C(C)C1)NC(=O)CCCCCF 11090,C1(C(N(C2CCCC2)CC=C)=O)CC2C=CC1N(C(=O)CC(=O)OC)C2 11091,CC1(C)C(NC(CC2(C(=O)NC3CCOCC3)CCC2)=O)CC1COC(C)C 11092,c1(C(=O)NC2C(CNC(C(COC)N(C)C)=O)CC2)cnn2ccn(C)c12 11093,C1(C)(N(C)C)CCN(C(c2cc(-c3c(Cl)cccc3Cl)on2)=O)CC1 11094,CCC(C(=O)N(CC(=O)NCC1(CCO)CN(C)C1)C1CC1)N(C)C 11095,N1(C(C(SC)SC)=O)CCC(CCC2CCCN2C(c2cnns2)=O)CC1 11096,n1(CC)nc(C(N2CCCC2CC(=O)N(C2CCC(O)CC2)C)=O)c(C)n1 11097,C(=O)(C1=CCCSC1)NC1C(CNC(c2ccc(CNC(C)=O)cc2)=O)CCCC1 11098,C(=O)(CCC(=O)N(CC)CC)N1CC(OCC)(CO)C1.C1(CC(=O)N)CCCN1C 11099,N1(C(CC(CNC(=O)COCCCN=[N+]=[N-])OC)=O)CCN(C)CC1C 11100,C(=O)(C#CC(C)(C)O)N1CCCC(NC(C(CC)(C)C)=O)C1 11101,C12(C(N3C(CC)CC(C)C3)=O)COCC1CN(C(C1CC1(C)C)=O)C2 11102,C(=O)(C(O)CC(C)C)NC1(CCNC(CNC(CCC(C)C)=O)=O)CCC1 11103,c1(C(=O)NCC(CCOC)NC(=O)C=C(C2CC2)C2CC2)ccc2snnc2c1 11104,N1(C(CCCOCC=C)=O)C2CCC1C(NC(=O)CNC=O)C2 11105,C1(CNC(c2c(C)c(F)ccc2)=O)CCCCN(C(=O)Cc2n[nH]c(=N)s2)CC1 11106,C1(C(=O)NCC(C)OCC#C)C2CC3C(C2NC(C2(CO)CCOC2)=O)C13 11107,C1(C)(CNC(C=NOC)=O)COCCN(C(=O)Cn2ncc(O)nc2=O)C1 11108,N1(C(C2(C)CSC2)=O)CCC(CCCNC(=O)CCN2CCCC2)CC1 11109,C(=O)(CN=S(C)(C)=O)N1C(CN(C)C(C2CC2c2ccncc2)=O)COCC1 11110,N1(C(CC(=O)OC)=O)CC=CC(NC(=O)CCc2cncc(OC)c2)C1 11111,CCC(CCCC(=O)NC(C)COC)NC(C1CCCC1F)=O 11112,N1(C(c2cc(C3CC3)no2)=O)CCCC(CN2CCN(c3cnccn3)CC2)C1 11113,C1(CNC(c2c(C)cco2)=O)C(C2CC2)CCN1C(c1ncc[nH]c1=O)=O 11114,c1(CC)nnc(CN(C(C(C2COC2)NC)=O)C)s1 11115,C=CCCCC(C(=O)NC(C=C)C(F)(F)F)NC(=O)CCNC(C)=O 11116,c1(C(N2CC(c3cn(C)nc3)OCC2)=O)cccc(OC(F)(F)F)c1F 11117,C1(CC(=O)N(C(C)C(=O)NC2C3CCCC23)CC)CCCC(C)O1 11118,c1(C(=O)NCC2CCC(NC(C3C(CCC)C3)=O)CC2)nccc2cccnc12 11119,C1(NC(C(CC)CC)=O)CCN(C(c2ccoc2)=O)C(c2ccccc2)C1 11120,CC(C)(CNC(=O)CCc1cncnc1)CNC(c1nn[nH]c1C(F)(F)F)=O 11121,Cc1cc(CCC(=O)NCC2CCCN2C(c2cc(C)c(Cl)s2)=O)cc(C)n1 11122,C1(NC(C(=O)NC2CC(C)OC(C)C2)=O)CCCCC12CCCC2 11123,N1(C(c2cc(C(=O)OC)no2)=O)CCC(C(C)NC(=O)C=C2CCC2)CC1 11124,c1(C(N2CC(CC(C)NC(=O)CSCC#N)C2)=O)nc2c(s1)COCC2 11125,N1(C(c2cnn(CC)c2CC)C(=O)NCC)CC2(CC=CC2)C1C(C)C 11126,c1(CNC(C2CCN(C(c3ccncc3N3CCCC3)C)C2)=O)ccc(F)cc1 11127,N#CC1CCN(C(=O)CC(CC2CC2)NC(C2CCS(=O)CC2)=O)C2(CC2)C1 11128,c1(C(=O)NC2C3CN(C(C4CCCN(C(CC)=O)C4)=O)C2C3)cnc(F)c(C)c1 11129,N1(C(C(CC=C)C)=O)CC(NC(=O)Cc2ccoc2)CC(C)C1 11130,C(=O)(CCC(=O)NN(C)C)N(C)CC1(O)CCN(C(C(CC#C)O)=O)CC1 11131,c1(C(N(CCNC(=O)COC2CCCCCC2)CC)=O)nc2c(s1)CN(C)CC2 11132,C1(CNC(Cc2c(C)cccc2)=O)CC2(CO1)CN(C(c1c(C)n[nH]c1C)=O)C2 11133,C1(O)(C(C)NC(COCCCC)=O)CCN(C(=O)CCc2nc[nH]n2)CC1 11134,c1(CC(C=C)O)cn(CC(F)CCNC(=O)C(C)(C)OC2CCCC2)nn1 11135,C1(NC(CC2(C)CCOC2)=O)CCCCC1CC(N1CCC(n2ccnn2)C1)=O 11136,c1(C(C)C(=O)Nc2nc(CCNC(c3ccccc3)=O)cs2)cccc(Br)c1 11137,N1(C(c2cc(CC)[nH]n2)=O)CCC(CNC(=O)C(C)SC)C(C)C1 11138,c1(OC)ccc(Br)cc1C(N1C(C(N2CC(F)CC2C(N)=O)=O)CC2CC12)=O 11139,N1(C(CC(C)N(C(C(C(=O)OCC)CC)=O)C)=O)CC2(C1)NC(=O)NC2=O 11140,c1(C2(C(C=O)N3CCCC3)CC2)cccc(F)c1.c1(C(C)O)ccccn1 11141,N1(C(C=Cc2ncn(C)c2)=O)C2CCC1CN(C(c1cc(C3CC3)sn1)=O)CC2 11142,c1(N2CC2=O)ccc(Br)c(Cl)c1.N12CCCCC1C2.C#CCCC1N=N1 11143,CCC(C)CC(=O)NC1CC(CNC(=O)CSCc2ccc(Cl)s2)C1 11144,c1(OC)nccc(C(=O)NC2CC(C(=O)N(C3CCN(C(C)C)C3)C)C2(C)C)n1 11145,N1(C(CCSC)=O)CCN(C(C23CCC(N=[N+]=[N-])C2C3)=O)C(C)C1C 11146,c1(OC)cc(C(=O)NC(C)CC2CN(C(=O)CN3CC4CC4C3)C2)sn1 11147,c1(OC)ccc(CC(=O)NCC2C=CCN2C(c2conc2C)=O)cn1 11148,c1(C(=O)NCC2(OC)CN(C(c3ncsc3C(F)(F)F)=O)C2)occ2c1CCC2 11149,C(=O)(C(C)(C)CS(N)(=O)=O)NCC1CN(C(C(CC)NC(C)=O)=O)CC1O 11150,Cc1ccc(C(=O)O)c(-n2cc(-c3ccns3)nn2)c1.C12CCCN(C1)C2 11151,N1(C(c2c(C)n[nH]c2C)=O)CCN2C(=O)C(NC(=O)CC(C)(C)C)CC2C1 11152,c1(OC)ccc(NC(c2ccccc2NS(=O)(=O)C2CC2)=O)c(OC)c1OC 11153,C(CC(C)C(=O)NC(C1CCN(C(=O)C(=C2CCCCC2)F)CC1)CO)OC 11154,C1(O)(C(C(=O)NOCCOCC2CCC2)NC(CN(C)C)=O)CCCCC1 11155,Cn1oc(C(=O)NC2CCCC2CNC(C23CC(C(F)F)(CO2)C3)=O)cc1=O 11156,c1(O)cc(Cl)ccc1Cl.C1(C(=O)NC2CN(CC)C2)(NC(C(C)O)=O)CCOCC1 11157,c1(C(NNC(C(=O)N(CC)CC)=O)=O)cn2c(n1)C(C)CCC2 11158,N1(C(CCC=CC)=O)CCCCCC(NC(=O)C(C(C)O)N(C)C)C1 11159,Cc1ccc(CC(=O)N(CCCCCNC(C2(F)CCOC2)=O)C2CC2)cc1 11160,C1(CNC(CC(=C)C)=O)CN(C(c2ccc(C(C)C)nc2O)=O)CCCO1 11161,CN1CCCCC1CC(=O)NC1CCCC1(C)CNC(c1c[nH]nc1C(F)F)=O 11162,c1(C(N(CCNC(=O)C(C)C)CC)=O)cc(OC)c2c(c1)OCO2 11163,C1(C(=O)NC2CCCN(C(C3(CN(C)C)CCCC3)=O)C2)CC(=O)NC1(C)C 11164,N1(C(CCC(C)(C)NC(=O)Cn2cnnc2O)=O)CC2CC(C1)C2(C)C 11165,c1(OC)ccc(C)c(C(=O)NCC2(CCCNC(=O)C=C(C)C)CCCC2)n1 11166,O=S(=O)(c1cccc(F)c1)NC1CN(Cc2ccccc2)CC2(CCC2)O1 11167,c1(OC)cc(C(=O)NCC2CCC2NC(c2cc(Br)n(C)n2)=O)ccc1C 11168,c1(C(N2CCC(N(C(=O)CC3CCC(=O)N3C)C)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 11169,c1(C(N2CCC(CC)C2C(=O)NCC2CC(C(C)C)C2)=O)ccc2n[nH]cc2c1 11170,c1(C(CC)NC(C)CC2CCCCO2)cccc(Cl)c1Cl 11171,c1(N(C)CCc2ccccc2)nc(=NCC2CCC3CC23)[nH]c2cccc(F)c12 11172,c1(C(N(C2C(O)CCN(C(c3nc(C)oc3C)=O)C2)C)=O)cccc2c1OCC2 11173,C(=O)(C(CC(N)=O)NC(=O)OC(C)(C)C)NC1C2(CC(NC)C2)C1 11174,Cn1cnn(CC(N2CC(CNC(=O)CCc3ccc(Cl)cc3)C2)=O)c1=O 11175,C1(C(NOCC=C)=O)COCCN1C(c1ccc(C)nc1)=O 11176,c1(C(=O)NC2(C(N(C(C)C(C)(C)C)C)=O)CCC(C)(C)C2)coc2ccccc12 11177,c1(C(N2C(COC)CN(C(=O)C=C(C)C)CC2)=O)cnn2ccc(OC)cc12 11178,c1(CC)cc(N(C)CC2(CNC(=O)C(C3CCOCC3)O)CC2)nc(CC)n1 11179,C1(C(N(CC(C2CC2)OC)C)=O)C2CCCC2CN1C(=O)Cn1ccccc1=O 11180,N1(CC)CC(NC(C2(NC(c3ncncc3Cl)=O)CC(O)C2)=O)CC1=O 11181,n1(CC(=O)NC2CC3CC2CN3C(c2ccoc2C2CC2)=O)nc(O)ccc1=O 11182,CCC(CNC(=O)C(=O)NC1CC(=O)N(C(C)C)C1)(CC)c1ccccc1 11183,Cc1c(C(=O)N(CCC(=O)NC(CO)CCF)C2CC2)ccn1C 11184,c1(-c2cn(CC3CCN(C(CN(C)C)=O)C3)nn2)cc(CO)ccn1 11185,CCC(C(=O)N(C1(C(=O)NCC(F)Cl)CC1)C)C(C)C 11186,c1(CC(=O)NC(C(C)NC(c2c(CC)ocn2)=O)(C)C)ccc(F)c(Cl)c1F 11187,C(CN=c1cc(C)c(S(=O)(=O)N2C(C)CCC2C)c[nH]1)SCC=C 11188,c1(C(C)N(C(C2CC3CCC2CC3)C(=O)NCC2CC2)C)nc2ccccc2s1 11189,C(CCN(C)C(c1ccns1)=O)(C(C)(C)C)NC(c1cccc(COC)n1)=O 11190,CN1CCCCC(C(=O)NCC(C)(C)CNC(C2(C)CCC(=O)C2)=O)C1=O 11191,c1(CCC)noc(CCC(=O)NC2CCN(C(=O)C=C(C)C(F)F)C2)n1 11192,C1(CNC(c2occ(C)c2)=O)CC(C)N(C(c2cn(C(C)C)cn2)=O)C1 11193,C(C)(CCC(C)(C)C)N(C(c1nn(C)cc1O)C)CCOCc1ccccc1 11194,CC(C)P(=O)(CC(=O)NCC1(C(C)(C)O)CN(C(=O)C(C)(C)F)C1)C(C)C 11195,C1(O)(CNC(CC2(N(C(CC3(OCC)CC3)=O)C)CC2)=O)CCCC1C 11196,CCCCC(CNC(=O)COCCCF)NC(=O)C(C)Oc1cccc(C)c1 11197,CC(=O)C(C)CC(C)C(=O)NCCCC(C)(C)NC(c1n[nH]c2c1CCOC2)=O 11198,c1(C(N(C)C)=O)cccc(F)c1-c1cncc(NC(c2ccncc2F)=O)c1 11199,c1(N(C)Cc2nnn(C(C)(C)C)n2)cccn2nnnc12.C12CC(F)CN1C2 11200,c1(C(=O)NCC2(CN(C)C(c3ccc(Cl)cc3)=O)CC2)cnn(C)c1N 11201,Cn1nnc2cccc(CO)c12.N12CCN(C1=O)C1CN(C1)C(=O)C2 11202,N1(C(C2(SC)CCC2)=O)CCN(C(C2CCCCS2)=O)C(c2nccn2C)C1 11203,c1(C(=O)NCCC2(CNC(CN(S(C)(=O)=O)C)=O)CC2)nnc2ccccc2n1 11204,c1(OCC)cccc(C(=O)NC2(C)CCN(C(c3n[nH]c(C4CC4)n3)=O)C2)c1 11205,c1(C(C(=O)NCCN(C(C(C)C2CCC2)=O)C)C)ccc(Cl)c(Cl)c1 11206,N1(C(C(C=C=C)C)=O)CC2CCN(C(c3nc4ncc(C)cn4n3)=O)C(C2)C1 11207,N1(C(CCC2(NC(COCCOC)=O)CCC2)=O)CCC(CO)C(C)(C)C1 11208,Cc1cccc(C(C(F)(F)F)NC(=O)Cn2cc(C(C)(C)S(C)(=O)=O)nn2)c1 11209,C(C(CCC)CCC)NC(CCC#CC)=O 11210,N1(C(CC(COC)C)=O)CCCC(C)(NC(=O)CCCc2ccc(Cl)cc2)C1 11211,N1(C(C2CCC(C(=O)OC)C2)=O)CC2CC(C)N(C(c3ccsc3Cl)=O)C2C1 11212,c1(CC)cc(C(=O)NCC2(C(N3CC(O)C3)=O)CC(C)(C)C2)c(C)o1 11213,C1(C(=O)NCC2(F)CC(CNC(C3CCCO3)=O)C2)Cc2ccccc2S1 11214,CCCCC(O)C(=O)NC(CCC(=O)N(CCO)CCN(C)C)C(C)C 11215,C(=O)(CCS(=O)(=O)C(F)(F)F)NCC1CCN(C(c2n(C)ncc2C2CC2)=O)C1 11216,CC1COCCC1NC(=O)C(CC1CCC1)NC(=O)CC=C(Cl)Cl 11217,C1(NC(c2cnc(CO)cn2)=O)CN(C(=O)CCOC2CCCC2)CCC1CO 11218,CC(C)CC(C(=O)N1CC(C(=O)NCCc2ncon2)CC(C)C1)C(N)=O 11219,CC(C)(C)C(CNC(=O)C(O)CC1CCOCC1)NC(C1(CF)CCC1)=O 11220,C1(NC(C2N(C(c3cc(CC)no3)=O)CC2C)=O)CC2(CCC2)C1OC 11221,N1(CCC(C)F)CCC2(CCN(C(=O)C(C)(C)C3CC3)C2)C1 11222,N1(C(C(CC)OC)=O)CCC(C(F)F)(CNC(=O)CCn2cccnc2=O)C1 11223,c1(NC(C2C3(CN(C(CC(CC)C)=O)C3)C2)=O)cc(F)c([N+](=O)[O-])cc1F 11224,c1(C(N(CC(CC)NC(C2(O)CCOC2)=O)C)=O)ccsc1SC 11225,c1(NC(=O)Nc2cncc(F)c2)ccc(S(=O)(=O)CC2CCCO2)cc1 11226,N1(C(Cc2c(C)ccnc2)=O)CC2CCC1C(NC(c1nc(C)n(C)n1)=O)C2 11227,C1(CNC(c2ncn(C(C)(C)C)n2)=O)CC2CCC1N2C(C1(C)CCC(=O)C1)=O 11228,C(=O)(C1CCCc2ncccc21)NCC(CNC(c1c(C)onc1C1CC1)=O)C 11229,c1(C2N(C(C3N(c4ccnc(OC)n4)CCCC3)=O)CCC2)ccc(Br)cc1F 11230,CC1(NC(c2ccccc2)=O)CC(NC(C2CC2(C)C(F)F)=O)C1 11231,C(N=c1cc[nH]cc1S(=O)(=O)NC(C)(C)C1CC1)c1cnc(CC)s1 11232,N1(C(C(CC)(C)CNC(C2CC2OC(C)=O)=O)=O)CCC2CCC(C1)N2C 11233,C1(C(=O)NCCC(C)N(C(C(C)OCC#C)=O)C)CC12CCOCC2 11234,CC(CNC(C1CC1)=O)CCC(=O)N(c1nccs1)CCO 11235,N1(C(C(C)N(CCC)C(C2CCCCS2)=O)=O)CC2(COC(=O)C2)C1 11236,c1(NC(C)=O)ccc(C(=O)NC23CCN(C(=O)OC(C)(C)C)CC2C3)c(C)c1 11237,c1(C(N(CCNC(C2N(C(C)=O)CSC2)=O)C2CC2)=O)cnc(C2CC2)nc1C 11238,C1(C)(CNC(C(c2cccnc2)C)=O)CCCN1C(c1cccc[n+]1[O-])=O 11239,c1(C(=O)NCC(C)NC(=O)C(c2ccc(Cl)cc2Cl)O)nccc2[nH]ccc12 11240,c1(C(=O)NCCC(C)NC(c2ccnc(S)c2)=O)ccc2c(c1)CCO2 11241,C(=O)(CC(O)CNC(=O)CCCN(C)C)NC(C1CSC1)C 11242,Cc1nc(N2CCC(NC(=O)Cn3nnnc3C)C(O)C2)cc(C#N)n1 11243,N1(C(C2(C)COC2)=O)CC(C(N2CCCCC2CCCO)=O)C(C)(C)C1 11244,C(=O)(CC1OCc2ccccc21)N1CC=C(CNC(C(C)OC)=O)CC1 11245,Cn1c(=N)[nH]c2ccc(C(=O)OC(C)(C)C)cc12.c12cnn(c1)CC(=O)N2 11246,C1(CC(=O)NCC(CC)OC)CCCN1C(c1csc(NC(=O)C2CC2)n1)=O 11247,c1(NC(C2C(CNC(C3CCC(C4CC4)C3)=O)OCC2)=O)cnc2c(c1)CCC2 11248,c1(C(N(CCCCNC(C2CC2C2CCCO2)=O)C)=O)ccncc1Br 11249,C1(NC(C(CSC)C)=O)CC2CN(C(c3cc(-c4ccncc4)[nH]n3)=O)CC12 11250,N1(C(C(Cc2cn[nH]c2)NC(c2cc(OC)no2)=O)=O)CCOCC1CC(C)C 11251,CC1(C2(C(=O)NCC(O)C(N3CCOCC3CO)=O)CC2)CC1 11252,N1(C(C(C)(C)NC(=O)C(F)(F)F)=O)CC2CN(C(C3CC(=O)C3)=O)CC2C1 11253,C1(N=[N+]=[N-])(C(=O)NCC(CCC)OC)CCN(C(=O)CCCC(C)(C)C)C1 11254,N1(C(c2nc(C)nc(O)c2)=O)CC2CCN(C(c3cc(C(F)F)n(C)n3)=O)CC12 11255,c1(NC(=O)NCCCN2C(C)CCCC2)nc2cccc(Cl)c2[nH]1 11256,C1(C(N(C(C2CCCCC2)C)C)=O)CCN(C(=O)C(C)(C)Br)CC1O 11257,c1(C(=O)OC)nccn1CC1CN(C(=O)CC2(NC(=O)C(C)(Cl)Cl)CCC2)C1 11258,N1(C(=O)CCC2CCOC2)CCCC2C1CCN2C(=O)C(F)F 11259,C(CC(F)(F)Cn1cc(C(CC)OC)nn1)NC(C1(CCCC)CC1)=O 11260,N1(C(CC2(C)CCN2C(=O)COC2CCOC2)=O)CCC2(CCCCC2)C1 11261,N1(C(c2cncc(C)n2)=O)CCC2CN(C(c3nc(C4CC4)cs3)=O)CC2C1 11262,C1(C(=O)NCCCN(C(=O)CC2CCCCO2)C)(CC)CCOCC1 11263,c1(CCC(=O)N(C2CCN(C(C3CC=CCO3)=O)CC2)CC#C)ccccc1C 11264,S(=O)(=O)(c1cccs1)N(CCCO)C.C12CCN(CC1)C(=O)C(=O)NCC2 11265,N1(C(CC(=C)C)=O)CC(NC(=O)CCc2cc(Cl)no2)CC(C)C1 11266,c1(C(N2C3CN(C(C4C(CCC)C4)=O)C(C3)C2)=O)ccc(Br)c2cn[nH]c12 11267,c1(C(=O)NCC2CCN2C(c2cc(Cl)cs2)=O)c[nH]c2nccc-2c1 11268,c1(NC(=O)NNC(=O)Cc2csc3ccc(Br)cc23)ccc2c(c1)CCCO2 11269,N1(C(C(C)=C(C)C)=O)CCC(NC(c2cc(C)cnc2Cl)=O)CC1C 11270,C1(CC)CCC(C(=O)NC2(C)CCN(C(=O)C(COC(C)C)NC(C)=O)C2)CC1 11271,c1(NCc2c(N)ncc(Br)c2)ccc(S(=O)(=O)NC2CCC=CCC2)c(Br)c1 11272,Cc1cc(C)cc(C=CC(=O)NC(C)C(C(C)C)NC(=O)CCC(C)(F)F)c1 11273,CC(C)(CCCF)C(=O)NCC1CCN(C(C2CCCC(=O)CC2)=O)C1 11274,N1(C(CC(CNC(c2c(C)cn(C)n2)=O)O)=O)CCN2CCCCC1C2 11275,N1(C(C(Br)=C(C)C)=O)CC(CNC(=O)COC2CCCCC2)CCC1C 11276,N1(C(c2cnc(C)o2)=O)CC(NC(c2ccc(CC(C)(C)C)cc2)=O)CC1C 11277,C(=O)(CCS(C)(=O)=O)N1CCC(CC)C1CNC(=O)C(=Cc1cccnc1)C 11278,C1(C(=O)NC(C)CCF)CN(C(=O)CCC2CC2(F)F)C2(CCC2)C1 11279,c1(OC)ncc(C=CC(N2CC(NC(C3CCCS3)=O)C3(CC3)C2)=O)cn1 11280,C=CC1(CC(=O)NC(C)Cc2ccnn2C)CN(C(=O)CCN(C)C)C1 11281,Cc1onc(Cl)c1C(=O)NC1CCN(C(c2ccc(C#N)s2)=O)C1 11282,C1(C(N2CCC(CNC(CCNS(CC)(=O)=O)=O)CC2)=O)CCCCC1(F)F 11283,N1(C(CC2C(C)C2)=O)CCCC2(CCN(C(c3cc(C4(C)CC4)on3)=O)C2)C1 11284,CC1CC=C(C(=O)N2CCC(CN(C)C(c3cccc(O)c3F)=O)C2)CC1 11285,Cc1cc2nc[nH]c(=NCC(C)NC(=O)C(c3ccc(F)cc3)CC)c2[nH]1 11286,C1(C(N2CCN(C(c3c(Cl)ccc(C)c3)=O)C(C)C2)=O)CCCC2CCCN12 11287,Cc1cc(NC(=O)CCc2ccc(C(=O)Nc3ncco3)[nH]2)nc(Br)c1 11288,C1(CN(C(C(C)O)=O)C)CCCN(C(=O)C=CCN2CCC2)C1 11289,c1(CN(CCNC2CCN(CC(F)(F)F)C(=O)C2)CC)ccc(O)c(Br)c1 11290,c1(NC(C(CNC(=O)CCNC(N)=O)OC)=O)cccc(C(C)F)c1 11291,c1(NC2C(C(=O)Nc3c(OC)cc(F)c(C)c3)C2)ncnc2c(C)cccc12 11292,CC1=C(C(=O)N(CCCCCNC(=O)C(F)C2CCOC2)C)SCCO1 11293,N1(C(CC2(O)CCCN(C(C)=O)C2)=O)CC2CN(C(c3c[nH]cc3Br)=O)CC2C1 11294,c1(C(=O)NC2C3N(C(C)=O)CC(CC3)C2)cc(N(C)C)nc2ccccc12 11295,Cc1cc(O)cc(O)c1NC(=O)C(C1CCN(C(=O)C(C)(O)C(F)(F)F)CC1)C 11296,c1(C(=O)NCC23C(CN(C(C(CC)COC)=O)C2)CC3)cnc2[nH]cnc2c1 11297,C1(N(C)C)CC(C(=O)O)CN(C(=O)CC2CC(SC(C)(C)C)C2)C1 11298,CC(C)C(O)C(C)C(=O)N1CC(C(=O)NC2CC(C3CC3)C2)CCC1C 11299,N1(C(COCCC)=O)CC(N(C(=O)CNc2cccnc2)C)C(C)(C)C1 11300,C1(C)(CNC(C2(CC=C)CC=CC2)=O)CCCN(C(=O)CN2CCCCCC2)C1 11301,C#CCC(C)(CNC(=O)NCc1cc(C(=O)OC(C)(C)C)c(C)s1)CO 11302,CC(CC(C)(C)C)C(=O)NCC12CCC(CN1C(c1cc(Br)n[nH]1)=O)C2 11303,N1(C(CC(C)F)=O)CCCC(CN2CCN(C(c3ccc(C(N)=O)s3)=O)CC2)C1 11304,N1(C(Cc2nc(C)oc2)=O)CC2ON=C(CNC(c3nnc(C)s3)=O)C2C1 11305,C12CC3CC(C3C1)NC2=O.c1(CC2CC(CC(=O)OC)C2)ccccc1 11306,C(=O)(C(C(C)(C)C)OCC)N(CCC)CCNC(C12CCCC1C2)=O 11307,N1(CC(N2CCC(C3CCCN3C(C34CSCC3C4)=O)C2)=O)CCC(F)CC1 11308,c1(N2CCCC(C(C)C)(CO)C2)nc(N2CCOC(C)(C)C2)c2cnn(C)c2n1 11309,c1(CC)ccc(C(C)NC(c2nnnn2C(C)(C)CC)(c2nccn2C)C)cc1 11310,C1(NC(c2c(CC)nc[nH]2)=O)(CC)CCN(C(c2ccoc2C2CC2)=O)CC1 11311,Cc1[nH]c(C(=O)NC(CCN(C(=O)C(N)=O)C)C(C)C)c(C)c1C 11312,CC1OC(C)C(C(=O)NC2(CCCCNC(=O)CC3CC(F)(F)C3)CC2)C1C 11313,c1(C(N(C2CCCN(C(C3CCCC3)=O)CC2)C)=O)cc(N)cc(O)c1F 11314,N1(C(C2CC(OC)C2)=O)CCCC(CN(C(=O)CN(C)C(=O)OC(C)(C)C)C)C1 11315,CC(C)C(CNC(=O)CC1CSC1)C(=O)NCc1ccon1 11316,N1(C(N2CC3(CC3CNC(=O)OC(C)(C)C)C2)=O)CC(C)(C(=O)O)CC1(C)C 11317,O=C(C#CC1CCCCO1)NC1CCC2CCN(C(=O)CCC3CC3(Cl)Cl)C1C2 11318,Cc1cn2c(n1)CCC(C(=O)NC1CC(CNC(c3ccc(C)s3)=O)C1)C2 11319,C1(N(CCNC(C(F)=C(C)C)=O)C(c2cc(C3CC3C)on2)=O)CCCCCC1 11320,N1(C(C(F)OC)=O)CCC(NC(=O)C(Cc2ccsc2)NC=O)CC(C)(C)C1 11321,Cc1ccnc(CNC(C2COCCN(C(c3ccncc3)=O)C2)=O)c1F 11322,C1(C(N2CCN(C(=O)C=C3CCSCC3)C(C3CC3)C2)=O)CC2CCC(C1)C2 11323,c1(C(=O)NC(C)CN(C)C(c2ccsc2)=O)ccc2sc(=N)[nH]c2c1 11324,N1(CCNC(=O)NC(c2sccc2Cl)CC2CCCCC2)CCS(=O)(=O)CC1 11325,Cn1nc(Cn2cc(Br)cn2)nc1SCCCn1ccnc1 11326,C#CC1(C(=O)NCCC2(C)CCCC2)CCN(C(C2CCC(OC)C2)=O)CC1 11327,CC1(C)CCCN(C(C2CC(=O)CO2)=O)C1CNC(C1CCC(=C(F)F)CC1)=O 11328,C(=O)(CCCCCCC(=O)N1CCC(NC(c2ccc(SC)o2)=O)C(O)C1)OC 11329,C12(NC(c3ccc(OCC)cc3)=O)CCCC1CN(C(c1occc1F)=O)C2 11330,n1(CC(=O)NC2C(C)CN(C(C3CC34CC4)=O)C2)cnc2ccccc2c1=O 11331,c1(C(N2C(C3(NC(CCC=CC(C)C)=O)CC3)CCC2)=O)ncc(Cl)cc1O 11332,Cc1cc(CN=C(NC2CCC2)NC2CC23CCC3)c(C)n1-c1ccc(F)cc1 11333,C=C(Cl)C(C)(C)C(=O)NCC1CC(CNC(C2CC2c2cccnc2)=O)C1 11334,C(=O)(C1=C(Cl)CCOC1)NCC1C(NC(C2CCCC(C)(C)O2)=O)CCCC1 11335,C1(OC)CC2CCC1CC2C(=O)NC1CCCC(NC(=O)CCC2CCOC2)C1 11336,C1(NC(C23CC(C)(C2)C3)=O)CCC2CC1CN2C(=O)Cc1ncncc1Cl 11337,C(C)(C)(CC(=O)N(C)Cc1ccccn1)N(C(C1C(C)C1C)=O)C 11338,c1(C(=O)NCCN(C(C)C)C(c2cc(Cl)cn2C)=O)nc2n(c1Cl)CCCC2 11339,N1(C(CN2CCCC(CC)C2)=O)CCC(NC(=O)Cc2ccsc2Cl)C12CC2 11340,N1(C(C2CN(C(N)=O)C2)=O)CCOC2(CCC(NC(C3CC=CC3)=O)CC2)C1 11341,c1(N2C(C3(NC(c4ccoc4Br)=O)CC3)CCC2)ccc([N+](=O)[O-])cc1 11342,CC(C)CC(C)C(=O)NCC(C)NC(c1c(Br)cnn1C)=O 11343,C(=O)(C1=CC2C=CC(C1)C2)NC(C(=O)N(C(C=C)C)C)CO 11344,C1(NC(C=NOC)=O)C2CC3CN(C(=O)CCCCC(F)(F)F)C1C3C2 11345,CCC(CNC(c1cscc1C)=O)(CC)NC(c1ccc(C2COC2)cc1)=O 11346,N1(C(c2nc(CC)oc2)=O)CCC2(COC(CNC(=O)CCS(C)(=O)=O)C2)C1 11347,Cc1ccc(CNC(=O)NC2C3CC3C3CC23)n1Cc1cccs1 11348,CCCC(C(=O)NC1(CO)CN(C(c2nc(C)oc2C)=O)C1)N(C)C 11349,N1(C(C=CCCC=C(C)C)=O)CC2(CCCC2)C1 11350,CCC(COC)C(=O)NC(C)CC(C)NC(c1ccn(CC)n1)=O 11351,O=C(CCc1ccco1)NCCN(C(=O)Cc1nc[nH]n1)CC1CC1 11352,C(CCS(=O)(=O)NCC(N1CC(NC(C2(C)CCCC2O)=O)C1)=O)OC 11353,CCC(CC)C(=O)NCC(=O)NCCCC1(NC(=O)C(C)C(C)O)CC1 11354,CC1=C(C)CC(C)(C(N2CC(F)(CNC(C3CC4CCC(C3)S4)=O)C2)=O)CC1 11355,n1(CC(=O)NC(CCOC)CNC(=O)Cn2ccc(C3CC3)n2)c(C)ccc1C 11356,Cc1ncc(F)c(N2CCC(C#N)(NC(c3n[nH]c(C)c3C)=O)C2)n1 11357,C1(NC(c2n[nH]cc2C2CCC2)=O)CC2(C1)CN(C(C1CCCCO1)=O)C2 11358,c1(C(=O)NC2CN(C(=O)C(F)(F)c3nccs3)CCC2F)cccc2nccn12 11359,N1(C(C(C)N(C)C)=O)CCCCC1CNC(=O)C(F)(F)c1cnn(C)c1 11360,c1(CCC(=O)NCC(C)(C2CC2)NC(C(CCC)OC)=O)ccc2ocnc2c1 11361,CCC1c2ccsc2CCN1C(c1cc(F)ncc1C)C(=O)NC(C)(C)C 11362,C(C(C)(C)C(=O)NC(C)CCCNC(=O)C(O)CCSC)OCC 11363,Cc1cc(CS(=O)Cc2c(Cl)cccc2Cl)cc(C(F)(F)F)c1 11364,Cc1cc([N+](=O)[O-])cnc1C(N1CCC(C2(NC(c3csc(O)n3)=O)CC2)C1)=O 11365,CN1CCCC1C=CC(=O)NCCN(C(=O)C=Cc1cscn1)C1CC1 11366,c12ccc(c(OC)c1)OC(=O)CC2.C(=O)(C(C)=CC(C)(C)C)N(CC)CC 11367,C1(C(N2C(CN(C(c3ccc(C(C)C)cn3)=O)C)CCC2)=O)C(C)OC(C)C1C 11368,C(CO)(C(=O)NCc1cc(C(N2CCC(c3nn[nH]n3)C2)=O)co1)N(C)C 11369,c1(C(N(CC(CC)NC(CC(=C)I)=O)C)=O)n[nH]c(C)c1O 11370,Cc1cc(Cl)cnc1C(N1CC(O)(CCc2cn(C3CCCCC3)nn2)C1)=O 11371,Cc1cc(F)c(CC(N2CCN(c3ncccn3)C(=O)C2)=O)cc1F 11372,c1(NC)cc(F)ccc1CNC1(O)CCC(C(=O)OC)CC1 11373,CCC(CC(=O)NCCC1CC(C)C1)N(C)C(c1cnsc1C)=O 11374,c1(CNC(Cc2cn(CC)nn2)=O)ncccc1CNC(C1CNC(=O)C1)=O 11375,CCC(C(=O)OC)N(C(c1cnn(CCCl)c1)C(=O)NCC(F)F)C 11376,C=CC1OCCC1C(=O)NCCOC1CN(C(=O)CC(O)CN(C)C)C1 11377,C=CC(C)(C)CC(=O)NCC12CC(NC(c3cc(CC)ccc3F)=O)(C1)C2 11378,c1(NC(=O)NC(c2ccnn2C)C)cc(C(N)=O)c2n1CCOC2 11379,NS(=O)(=O)CC(=O)NCC1CN(C(=O)Cc2sccc2Cl)C1 11380,Cc1ccc(C(=O)NCCN(CC(C)O)C(c2coc(Br)c2)=O)o1 11381,c1cccc(Cl)c1.C1(C(=O)OCC)CC(F)(C(=O)NC2CC(CCNC=O)C2)C1 11382,C1(c2cn(Cc3ccc(C)o3)nn2)COCCN1C(=O)Cc1cn[nH]c1 11383,c1(OC)cc2[nH]ncc2cc1NC(=O)CC1CCN(C(c2cncnc2)=O)C1 11384,c1(NC(=O)OCC2CCCC2C(=O)NCC)ccc2c(c1)OCCO2 11385,Cc1cnc2n1CCCC2C(=O)NCCC1CC1C1CC1 11386,c1(C(N2CC(O)(Cn3cncn3)C2)=O)ccc(CNC(C2CC(O)C2)=O)nc1 11387,N1(C(=O)CCn2cncn2)CC(O)C(O)C1CNC(C1(O)CC1)=O 11388,C1(C(=O)NCc2occ(C(=O)NC3C(C)CCC3C)c2)CC(=O)CC(=O)N1 11389,N1(C(C2CCC(=C)CC2)=O)CCC2CCN(C(=O)C(C)SC(C)C)CC2C1 11390,c1(C(N2CC(NC(c3ccc(O)nn3)=O)CC(C)C2)=O)cc2c(cn1)OCCO2 11391,c1(C(CCc2ccccc2)NC(C(c2cccnc2)OCC)=O)nc(C)n(C)n1 11392,C(C#CC(F)(F)F)NC(C1CCN(C(C(=O)NC)=O)C1)=O 11393,c1(NC2CCC(NCC(Br)=C(C)C)C2)ccc(S(=O)(=O)N(C)C)cc1C#N 11394,c1(C(=O)NC2CCCN(C(C3CCCC34CC4)=O)C2)ccc2c(c1)C=CS2(=O)=O 11395,c1(-n2cc(Cn3cnc(C(=O)OC)n3)nn2)cccc(OCc2cscn2)c1 11396,Cn1c(C(N2CCOC(C3CN(C(=O)C=CCO)C3)C2)=O)cnc1O 11397,C(N=c1cc(C)nc(NC(C)C(C2CCCCC2)C)[nH]1)C1(OC)CCSC1 11398,C(CCC(C)C)(C(=O)NCc1ccc(OC(F)F)cc1F)NC(C)=O.C1CO1 11399,c1(NC(C2CC(C)CN2Cc2cncc(O)c2)=O)ccc(C(N)=O)c(F)c1 11400,C1(NC(CC(=O)OCC)CC#N)CC2COCC(C1)C2 11401,c1(C(=O)NCC(CO)NC(c2ccc(C3(C)CC3)cc2)=O)cccc([N+](=O)[O-])c1 11402,Cc1c(Cl)ccnc1C(N1CCC(CF)(NC(=O)CCc2ncc[nH]2)C1)=O 11403,c1(C(=O)Nc2cc(C(C)O)c(F)cc2)nc(O)c2ccccc2n1 11404,n1(CC(C)NC(=O)CC2CCOC2)cc(C(C2(c3ccccn3)CC2)C)nn1 11405,Cn1nccc1C1CC1NC(N1CCC(c2ncccn2)C1)=O 11406,N1(C(=O)Nc2n(C)c(=O)on2)CCN2C(=O)COCC2C1 11407,C(N=c1[nH]cnc2cc(C)[nH]c12)C1C(N(C(=O)CN2CCCC2=O)CC)CCC1 11408,N1(C(C(CC)C)=O)C2CCC1C(CNC(=O)Cc1ccccn1)C2 11409,c1(C(=O)NC2(CC(NOC3CCN(C)CC3)=O)CC2)cccc2[nH]ncc12 11410,C12(C(N3CCCC(N(C(C4CCN(C)C4=O)=O)C)C3)=O)CCC(CC1)CO2 11411,C1(NC(C(C)SCCCC)=O)CN(C(c2cc(CCOC)on2)=O)CC1C 11412,Cc1cc(C)c(CC(N2CC3CCC2C(C(=O)NCC(F)CO)C3)=O)c(C)c1 11413,C1(C(=O)NCCN(C(=O)C2=CCCOC2)CC(C)O)C(C)(C)CCCC1(C)C 11414,N1(C(c2c(CC)c(C)sc2)=O)CCCC2(C1)CN(C(C1CN3CCN1CC3)=O)C2 11415,Fc1cccc2cccc(CNCc3cc(F)cnc3Br)c12 11416,Cc1ccc(C(=O)NCC=CCNC(=O)C(=Cc2c[nH]cn2)F)cc1F 11417,C(C(C)(C)C(=O)NC(c1cccc(F)c1)C)N(C(c1ccc(CC)[nH]1)=O)C 11418,C(C(C)(COC)C(=O)N1CCC(NC(=O)CC2CSC2)C(CO)C1)OC 11419,N1(C(C2C(C(=O)OCC)C2)=O)Cc2ccnn2CC1C.C1(=O)CCCC(C)(C)N1 11420,Cn1cnc(CCNC(C2(C3CCCN3C(=O)CNc3cnn(C)c3)CC2)=O)n1 11421,C1(CNC(C2(COC)CCCC2)=O)CC(C)(C)CN1C(=O)C1CC1 11422,c1(C(=O)NCC(CCCC)NC(=O)C2=CCCC2(C)C)ccc(Cl)c(C)c1N 11423,C(=O)(CCC(F)(F)c1ccc(Br)cc1)NCCC(CC)F 11424,S(=O)(=O)(c1cccc(F)c1C)N1CCN(C2CN(C(C=COCC)=O)C2)CC1 11425,C(CCCCCC(=O)N1CC(CN)(CNC(=O)CC2CN3CCN2CC3)C1)SC 11426,C1(CNC(=O)COC2CCCNC2=O)CCNC2(CC2)C1 11427,CN1CCCC1C(N1CC(c2cc(C(F)(F)F)on2)C1)=O 11428,c1(C2(C(N(C3CN(C(=O)CCc4cn(C)cn4)C3)C)=O)CC2)ncccc1F 11429,C1(C(C)C(=O)N(C2(C(=O)NC(C)C(=O)NC3CC3)CC2)C)CCC(=O)N1 11430,c1(OC)ncc(Cl)cc1C(=O)NC1CCN(C(=O)C(C)C(F)F)C1 11431,C#Cc1cccc(N(c2nnc(CC(C)(C)C)n2Cc2cccc(C)c2C)C)c1 11432,N1(C(C)=O)CCN(C(C2(F)CCN(CC3CCCN3C)C2)=O)CC1 11433,C#Cc1ccc(C(F)(F)F)nc1NC(c1ccc(C=O)[nH]1)=O 11434,c1(NC(c2ccoc2)=O)ccsc1C(=O)NCCF 11435,c1(C(=O)NC(c2ccc(C)cc2)c2c(C)noc2C)cc(Cl)ccc1C 11436,C=C(C)C1OCCC1C(N1CCC2(CC2NC(c2ccc(CO)o2)=O)C1)=O 11437,N1(C(c2cc(CC)ncc2)C(=O)NCc2cccs2)CCC(C2CC2)(CO)C1 11438,c1(OCC)ccccc1NC(=O)C(N1CCC(C)(CNC(C2CC(C)C2)=O)C1)=O 11439,N1(C(CC2N(C)CC=CC2)=O)CC2(CCCC2NC(c2ccc(=N)[nH]n2)=O)C1 11440,c1(N(C)Cc2cn(C)nn2)ccc(S(=O)(=O)NC2(C3CCSCC3)CC2)cc1F 11441,C(=O)(C(CC)C(=O)OCC)N(CCN(C(c1nccc(CC)c1)=O)C)C 11442,CC1=C(C(=O)NC(C)C(C)NC(c2cc3c(C)cccn3c2)=O)C(=O)OC1(C)C 11443,C1(C)(NC(C2(C(C)(C)OC)CC2)=O)CN(C(=O)Cc2cnc(C(C)C)o2)C1 11444,N1(C(COC)=O)CC2(C(=O)NC(C)CCC3CC3)CC1CCO2 11445,c1(C(C(=O)NCCC2(NC(C3CC34CCC4)=O)CC2)(F)F)ccccc1F 11446,c1(CNC2CC(CC(=O)NCc3cccc(C(=O)OC)c3)C2)c(I)ccnc1Cl 11447,C1(C(=O)NCC(C2CCC2)OC)CN(C(=O)C(O)CSC)CCC1(C)C 11448,N1(C(COCCCOC)=O)CCOCC1CNC(c1conc1C(C)C)=O 11449,C12(C(=O)NC(CC(=O)NC(C)C)C)CCC(CN(C(=O)C(CO)N(C)C)C1)C2 11450,N1(C(C=CC=CC)=O)CCOC(C(C)NC(=O)C(C)(C)c2ccccc2)C1 11451,n1(CCN(C)C)cc(C(=O)NC2CC2NC(c2cn(CC(F)(F)F)nn2)=O)nn1 11452,C12(C(=O)OCC)CCC1(C(=O)OC)CN(C(=O)NC1COC(C)(C)CO1)C2 11453,c1(SCC)ccc(CC(=O)NC(C)Cn2cc(-c3cnn(C)c3)nn2)cc1 11454,CCC(C)CC(C(=O)NCc1cccnc1)NC(c1cc(C(C)=O)[nH]n1)=O 11455,N12CCC(CC1)CC1(CC(=C)C1)NC2=O.N1(OC(C)(C)C)CCCC1 11456,N1(C(C2CC2C(=O)OCC)=O)CCCC2(C1)CN(C(c1ccnc(OC)c1)=O)C2 11457,C(C)(C)(CCCC(=O)N1CC(CC(C)C)C1)NC(c1cc(COC)on1)=O 11458,CCC(C(F)(F)F)NC(=O)C(=O)N(C1CCC1)C 11459,N#CC1CCCCC(C(=O)NCCN(CCOCCO)C(c2ccc[nH]2)=O)C1 11460,n1(COC)ccc(C(=O)NCC(C)N(C)C(C2CC2(F)F)=O)n1 11461,CC1CN(C(C2(C)CCCN2)=O)CCCN1C(c1cc(Cl)ccn1)=O 11462,C1(CC#C)(C(=O)NC2CN(C(=O)C=Cc3ccoc3)CC2OC)CCCCO1 11463,C(=O)(C(C)(CC)C(F)F)NC(CN(C(c1coc(C)n1)=O)CC)C 11464,C1(C2(O)CCCOC2)(NC(=O)NCCC2N(C(=O)OC(C)(C)C)CCOC2)CC1 11465,Cc1cc(C(=O)NC2CCCC(NC(c3ccsn3)=O)C2)ncc1S(N)(=O)=O 11466,C1(CC)CC(C)CN1C(c1c(Br)ncn1C)C(=O)NC(C)C(=O)OC 11467,N1(C(c2c(C)onc2)=O)CCC2(CC1)CC(C)N(C(c1ccc(CO)cn1)=O)C2 11468,CC1(C)CCc2c1n[nH]c2C(=O)NC1CCSC12CN(C(=O)C1CC1)C2 11469,N1(C(Cn2cc(C(N(C)C)=O)nn2)=O)C2CCCC1CC(NC(=O)CCCF)C2 11470,N12CC3CCC1C(C3)CNC(=O)C1(CCCC1)CC2.c1ncccc1C#N.CO 11471,c1(CN2CCC(NC(CCCCCCC)=O)(CO)CC2)cc2c(C)cccc2[nH]1 11472,Cc1nc(C#N)c(NCCC(=O)N(C2CCCCCC2)CCNC(=O)CO)o1 11473,N1(C(C(CO)NC(C(C)C)=O)=O)CCC(F)(CNC(=O)Cc2ccccc2F)C1 11474,N1(C(C(CNC(c2cncc(CC)c2)=O)CC2CC2)=O)CCCCCC1C 11475,C1(NC(c2csc(C(F)F)c2)=O)CC(NC(c2ccc[nH]2)=O)C12CCC2 11476,c1(CC)cc(C(=O)N(CCn2cc(C(C)(C)N(C)C)nn2)CC)c(C)nn1 11477,CCC(CC)(CC(=O)OC)NC(c1ccc(C(F)F)cc1OC)=O 11478,N1(C(Cc2cccc(SCC)c2)=O)CCC(NC(=O)C2=COCCO2)C(F)C1 11479,c1(C(N(c2ccc(Br)cc2)C(C)C)=O)cc(Br)c2[nH]c(=N)sc2c1 11480,N1(C(c2n(CC)ccc2)=O)CCCCCC1CNC(=O)C1=CCOC1 11481,C1(C(=O)O)CC(O)CN1c1ccc(C(F)F)nn1 11482,C1(C(=O)NCC(CCC)NC(c2cnns2)=O)(CC)CCOCC1 11483,C(=O)(C1Cc2ccccc21)N(C)CC1N(C(CCC=C=C)=O)CCOC1 11484,C1(C(=O)NC(C)CF)CN(C(c2cncc(N(C)C)c2)=O)CCC1(F)F 11485,N1(C(C2(CNC(c3ccc(NC)cn3)=O)CCCC2)=O)CCC2CN(C)CC12 11486,C1(OC)CN(C(=O)C=CC2CCCC2)CC1C(=O)NCC1CC(C)=NO1 11487,c1(CN(C(C2CC(CCNC(=O)CCCc3ncco3)C2)=O)CC)cccnc1 11488,c1(C(N2C3(CNC(C=CCC)=O)CCC2CC3)=O)ccc(Br)c(F)c1C 11489,C#Cc1ccc(C(=O)NC2(C(=O)NC(c3ncn(C)n3)C)CCSC2)cc1 11490,C1(COC)(CNC(c2nocc2C)=O)CCN(C(C2CCC(C)(C)C2)=O)C1 11491,C#Cc1cc(C(=O)NC2CCCC(NC(c3cnsc3)=O)C2)cc(Cl)c1 11492,n1(CC(CC)CC)nc(-c2ccc(C(C)C)cc2)nc1C1CCC(=O)N1C1CC1 11493,C(=O)(C(F)C(C)(C)O)NCC(C)N(C(=O)CSCCC#N)CC 11494,C12(CNC(c3c(CC)nc(C)nc3)=O)CCCC(CN1C(=O)CS(C)(=O)=O)C2 11495,c1(C(=O)OC)sc(C(N2CC=CC(NC(C3(N(C)C)CCCC3)=O)C2)=O)cc1N 11496,Cc1cc(Br)cc(C)c1NNC(=O)CNc1ccnc(F)c1 11497,c1(C(=O)NC2(CF)CCN(C(c3c(C)cnn3C)=O)C2)cncc(C)c1O 11498,Cc1cccc(F)c1C(N1CCC(C)(CNC(=O)CC(F)(F)Cl)CC1)=O 11499,N1(C(CC(C)(C)O)=O)CCC(NC(=O)CCNC(=O)CO)C(F)C1 11500,C1(C(N(CCOC)CCNC(c2coc(CF)n2)=O)=O)CC2OC(C)(C)OC2C1 11501,N(C1CCc2cccnc21)C(C(C1CCCO1)NC(CSCC=C)=O)=O 11502,c1(CC)cc(C(=O)N(CCCNC(=O)CC2CCC(C)C2)C)no1 11503,S(=O)(=O)(c1ccc(N(C)CCC2CC2)cc1Br)N(C(C)CN)C 11504,C1(CCNC(=O)CO)(NC(CC2CN(C)C2)=O)CCCC1 11505,C1(CNC(CN(CCCCCC)C)=O)CCCC(NC(=O)CS(N)(=O)=O)C1 11506,c1(C(N(CC(CN(C(c2c(CC)nc(C)o2)=O)C)O)C)=O)cccc(F)c1C 11507,c1(OC)cc(C(=O)N(CCC(C)NC(=O)C(O)Cc2cn(C)cn2)C)[nH]n1 11508,c1(C(N2C(C(=O)Nc3ccc(F)c(I)c3)COCC2)=O)cc(O)c(Br)c(O)c1 11509,CCCCC(CNC(=O)CC1CSC1)NC(c1n[nH]c(C)c1Cl)=O 11510,c1(OC)c(F)cc(CN2CC3CN(C(C4(OC(C)=O)CC4)=O)CC23)cc1F 11511,C1(N2CCN(CCOC)CC2)COC2(CCN(C(C3CCCO3)=O)CC2)C1 11512,N1(C(CC(=O)OCC)=O)CCC2(C=C(C(=O)N3CCOC(C)CC3)C2)C1 11513,C1(N=[N+]=[N-])(C(=O)NC(C(C)SC)C)CCN(C(c2oc(C)nc2C)=O)C1 11514,C1(NC(CC(CNC(c2ccnn2CCF)=O)O)=O)CCCCCCC1O 11515,c1(CC)nc(C)c(C(=O)NCCN(C(=O)C(C)C2CCC2)Cc2ccccc2)s1 11516,C1(CC)CC(C(=O)NC(CNC(=O)CC2CCOC2(C)C)C(C)(C)C)CCO1 11517,Cc1cnc(C(N2CC(CNC(c3cc(Cl)cnn3)=O)CC2C)=O)cc1Cl 11518,N1(C(c2ccnc(OC)n2)=O)CCCC2C1CCCN2C(=O)Cc1cc(C)ns1 11519,CCCC(CCC)C(C)NS(=O)(=O)Cc1ccc(F)cc1Cl 11520,N1(C(CN(C)C2CC2)=O)CCCC(O)(CNC(c2ccnnc2O)=O)C1 11521,c1(C(=O)NCCCCSC)occc1CNC(=O)C=CC(C)(C)C 11522,C1(C)(C(=O)NCC2C(C(N(CC(=O)NC(C)C)C)=O)CCO2)CCC(=O)CC1 11523,N1(CCC)CC(C(=O)NCCCCCCNC(c2ccsc2C)=O)CC1=O 11524,CC1CN(C(C2CC2CF)=O)CC1NC(C1CCC(N2CCCC2=O)CC1)=O 11525,C(=O)(CC1=CCOCC1)NC1(CO)CCN(C(C(C)Cc2cccnc2)=O)C1 11526,C(C)(CCCCNC(C1CCCC1(F)F)=O)NC(Cn1ccc(C(=O)OC)n1)=O 11527,N1(Cc2nccc(C)c2)CC(C(=O)Nc2ncc(CO)cc2Br)CC(F)C1 11528,CN1N=C(CC(=O)N2CCCCC(N(C)C(C3CC4(CCCO4)C3)=O)C2)CC1=O 11529,N1(C(c2cc(CC)ncc2)=O)CCCC(F)(C(=O)NCC(C)OCCOC)C1 11530,CC(C(C)(C)NC(c1cc(CO)[nH]n1)=O)NC(c1cnn(CC(F)(F)F)c1)=O 11531,C(CC1=CCN(C(=O)C(N2CCCCCC2)C)CC1)NC(C1C(=C)C1)=O 11532,C1(CNC(CC2CCC(=O)NC2)=O)(NC(c2csnn2)=O)CC2CCC1CC2 11533,c1(C(=O)NC2C(C)N(C(=O)CSC(F)F)CC2)c[nH]c2cnccc12 11534,N1(C(Cc2c(C)scc2)=O)CC2CC2(NC(=O)CCc2cncc(O)c2)C1 11535,C1(CNC(c2nc(C(C)C)sc2)=O)CCC(CNC(=O)CCc2ccc[nH]2)CC1 11536,C12(C(N(C)CC3CCN(C(C4C(C)(C)OC4(C)C)=O)C3)=O)CCCC(C)(C1)OC2 11537,C1(O)(C(=O)NCC2C3CN(c4nccc(C(C)=O)n4)CC32)CCCC(C)(C)CC1 11538,O(NC(=O)CC1(CNC(=O)COC(C)C)CC1)CC(C)C 11539,Cc1cn2c(CC(=O)NC(C)C(C)(C)NC(C3CCCCC(=O)N3)=O)csc2n1 11540,C1(NC(c2ccc(Br)s2)=O)CN(C(C2C=CC=CC=C2)=O)CC12CC2 11541,c1(C(=O)NCC(C)(CC)NC(CC(C=C)(C)O)=O)cnc2ncnn2c1O 11542,Cc1ccc2ccccc2c1NCC1CC(O)(CO)C1 11543,C1(NC(C2CN(C(C)=O)C2)=O)CN(C(C2(C)CC2(C)C)=O)CC1c1ccnn1C 11544,c1(C(=O)NCCC2CSCCN2C(=O)CC2CCOC2)cccc(C2CC2)c1F 11545,c1(C(=O)Nc2c(C)nc(C#N)cc2)n[nH]c2cc(C)ccc12.C(C)(C)(C)NC=O 11546,Cc1ccnc(C)c1CNC(c1coc(CNC(C2CC(F)C2)=O)c1)=O 11547,C(C(C)CC(=O)NC1CC(NC(c2coc(-c3ccccc3C)n2)=O)C1)OC 11548,c1(CC(=O)OCCCC)cccc(NC2CCCCC2CCCC)c1 11549,N1(C(C2CC2[N+](=O)[O-])=O)CCC(CNC(c2conc2C(F)(F)F)=O)CC1 11550,c1(C(=O)NCC(CCCC)NC(=O)C(F)C2CCC2)cnc2c(C)cccc2c1 11551,N1(C(Cc2nc(C)c(C)[nH]2)=O)CCC2CCCC12CNC(c1ccc(F)s1)=O 11552,N1(C(c2n[nH]c(=N)[nH]2)=O)C2CCC1C(C(=O)NCCC1CCCC1)C2 11553,C1(F)(C(N(CCO)CC)=O)CCN(C(=O)C(C2(O)CCCC2)F)C1 11554,C(=O)(NNc1cc(Cl)nc(N(c2cc(Cl)nc(Cl)c2)C(C)=O)n1)OC(C)(C)C 11555,C1(NC(C2CCCCC2)=O)CC2(C1)CC(NCc1cc(Cl)c(Cl)cn1)C2 11556,N1(c2cc(C)[nH]c(=NCC3CN4CCN3CC4)n2)CC2(C)CN(C)CC2(C)C1 11557,C1(CN(C)C(c2cnc(O)n2C)=O)CCC(NC(c2ncoc2Br)=O)CC1 11558,C1(C(N(CCCCC)C)=O)CCN(C(C23C=CC(CC2)C3)=O)CC1 11559,C1(C(=O)NCCN(C(=O)OC)C)COCCC1NC(c1ccccc1C)=O 11560,N1(C(C=CC)=O)C(CNC(=O)C(c2ccc(Br)cc2)OC)CC2CCCC12 11561,C#Cc1cc(F)c(C(=O)NC(C(C)NC(=O)CC(=O)NCC)C(C)C)cc1F 11562,C(=O)(C1CCCc2ncccc21)NC(CCSC)c1cccs1 11563,Cc1cncc(-c2cn(CC(=O)NC3C(C)=NOC3C)nn2)c1 11564,C(C(C(=O)NCCCn1ccnc1)NC(=O)C(N1CCCC1C)C)OC(C)C 11565,Cc1ccc(C(=O)NC2(CO)CCN(C(=O)C(C)(O)C3CCC3)C2)cc1Cl 11566,C1(NC(C(CC(=C)C)C)=O)(CNC(=O)CCC2CCC2)CC2CCC1CC2 11567,c1(OC)cc(C(=O)NCCCNC(=O)CSC(C)(C)C)c(F)cn1 11568,N1(Cc2nnc(CC)o2)CCCC(NC(=O)CCCOC(C)C)C1C 11569,C(C)(C(CC(=O)NCC1CC(SC)C1)NC(=O)C(C)NC=O)OC 11570,C12(CNC(C34CC(C(C)(C)C)(C3)C4)=O)CC(CN1C(C1(C#N)CCOC1)=O)C2 11571,c1(N2CCN(C)C(=O)C2)nc(=NCC2(CO)CC3CC3C2)[nH]c2cccnc12 11572,CC1(C2(C)CC2NC(=NCCC2(c3cccs3)CCC2)NC2CC2)CC1 11573,C12(NC(=O)CC=CCNC(=O)C(O)c3ccsc3)CC(CO)(C1)C2 11574,CC(C)(CCNC(C1CNC(=O)N1)=O)NC(=O)CCCc1ncco1 11575,c1(C(N2C(CNC(c3cnc[nH]3)=O)CCCC2)=O)cc2ccc(Cl)cc2c(=O)o1 11576,C1(COC(=O)CCOC2CCCCC2)CC2(CCC2)CN1C(=O)C1=COCCC1 11577,C(=O)(CCCCCN(C1CC2CC2C1)Cc1ccccc1)NC(C)(C)C 11578,c1(NCc2n(C)c(Br)nn2)[nH]c(=NCC(Cl)(Cl)Cl)nc2c1cnn2C 11579,Cc1nn(C)c(C(=O)NCC(C)NC(C2CC2c2cnn(C(C)C)c2)=O)c1Cl 11580,N1(C(C(COCC)OC)=O)CCC(N(C(=O)COCC(C)C)C)CC1 11581,c1(OC)cnc(CNCCN(C2CCCC2)C(=O)C=Cc2ncc[nH]2)nc1 11582,c1(C(N2CC(NC(CCN(CCCCC)CC)=O)C(C)C2)=O)cc(=O)cc(Cl)[nH]1 11583,c1(OC)nccc(C(N2CCN(C(=O)C(Cl)=CCl)CC2CS(C)(=O)=O)=O)c1F 11584,CC(C)CC(C(=O)N1CCCC1Cc1ccccc1)NC=O 11585,c1(CC(C)C)c(C(=O)N(C2CCC(NC(C34CCC3CC4)=O)C2)C)cnn1C 11586,N1(C(CC2N(C)CCOC2)=O)CCC2CN(C(c3nnn(C)c3N)=O)CC2CC1 11587,Cn1nc(Cl)cc1C(=O)NCC1(CNC(C2CC(F)C2)=O)CCCCC1 11588,C1(C)(NC(CC(C)C)=O)CCCN(C(=O)C(O)CN2CCCC2)C1 11589,c1(C(=O)NCCC(C)NC(C2CCCC(=O)CC2)=O)c[nH]cc(Cl)c1=O 11590,Cc1ccc(C(N2CCC(NC(c3ccncc3)=O)CC2C)=O)cc1OC(F)F 11591,CC1(C)CC(=O)OC1CNC(C1C=CCN(C(C2CCSCC2)=O)C1)=O 11592,C(CC(O)CC(=O)NC1COCC1NC(=O)CCCN(c1ccccc1)C)SC 11593,c1(C(=O)NC2CC3CN(C(C4(C)CC4(F)F)=O)C2C3)ccc(Cl)c2ncccc12 11594,C1(C(=O)NC2C(O)CCN(C(CCNC(=O)NC)=O)C2)CC2CCCCCC12 11595,CCC(C(=O)NC1(C)CC(NC(=O)CCC2CCCOC2)C1)N(CC)CC 11596,Cc1[nH]c(C(=O)NCc2ccc(F)cc2F)c(C)c1C(=O)NCC1CCCN1C 11597,N1(C(CC2(C)CC2)=O)CC(C)(C)OCC1CNC(=O)Cc1sccc1C(=O)CO 11598,N1(c2c(Br)cnc(C)n2)CCC2C1CCCN2C(c1c(Cl)cccc1Cl)=O 11599,c1(CC)ncc(C(=O)NCC2CC(F)(F)CN2C(=O)CN2CC3CC3C2)c(O)n1 11600,N1(C(CC2(C#N)CC2)=O)CCCC2CCCCC12.C12CCOCC1C(=O)N2 11601,N1(C(c2ccc([Si](C)(C)C)s2)C(=O)NCCCC)CCC2(C1)NC(=O)N(C)C2=O 11602,c1(COC)ccc(C(=O)NC2CCN(C(=O)CCCN3CCCC3)C2CO)cc1 11603,C1(CC(N2CC(CCNC(c3[nH]c(C)nc3C)=O)(OC)C2)=O)CCCNC(=O)C1 11604,Nc1cc(Cl)nc(Cl)c1C(N1CC2(COC(CNC(=O)Cc3cnoc3)C2)C1)=O 11605,Cc1ccc(C=CC(=O)NC(C2(O)CN(C(c3cnc(Cl)[nH]3)=O)C2)C)cc1Cl 11606,C1(O)(CNC(CC(CC)c2ccccc2)=O)CCN(C(c2ccc(=N)[nH]n2)=O)CC1 11607,C(=O)(C1CCc2ccccc21)N1CC2C(NC(C(CC=C)OC)=O)(CCC2)C1 11608,C(=O)(CCCCN1CCCCC1)NCCN(C(C(CC)O)=O)C1CCCCC1 11609,c1(C(c2nnnn2C)NCC2(OC)CC2)cc(Cl)nc(Cl)c1 11610,C1(NC(c2nnnn2C2CC2)(CSC)C)CCc2nncn2C1 11611,C1(CC=C)(C(=O)NC(C)CCC(=O)OC)CCN(C(=O)C=C(C)C(C)(C)C)C1 11612,N1(C(c2[nH]c(=NC)sc2)=O)CCC2CC2(NC(=O)CC2CCOCC2)CC1 11613,CCC(CC)C(=O)N(CC(C)NC(c1cnn(C(C)(C)C)c1CC)=O)C 11614,C(CC)(CC(C)CC)(c1n(CC(=C)C)nnn1)Nc1cc(SC(F)F)ccc1C 11615,c1(C(=O)NC2CC(NC(c3c[nH]c(=NC)s3)=O)C2)cccc(S(=O)(=O)C(F)F)c1 11616,C1(C)(NC(C=CC(C)NC(COC)=O)=O)CCC(C)=C(C)C1 11617,O=C(CCC[N+](=O)[O-])NC1(CCCN(C(=O)COC(=O)CO)CCO)CC1 11618,c1(CC(=O)NC(C(C)NC(c2c(COC)nn[nH]2)=O)C)ccc(F)cc1 11619,C(CCCCCCCCCCCO)NC(C1C(NC(c2cccs2)=O)C1)=O 11620,C=CC1CN(C(c2n[nH]c(C)c2C)=O)CC1NC(c1ncoc1C1CC1)=O 11621,c1(C(=O)NC2(CCCNC(C(C)n3cnnn3)=O)CC2)ccc(Br)nc1N 11622,N1(S(CC)(=O)=O)CCC(C(=O)NC(C)CCN(C(=O)CN(C)C(C)=O)C)CC1 11623,N#CC1(CC(N2CCCCCC2CNC(=O)C(F)n2cccn2)=O)CCOCC1 11624,CC1(C)CN(C(c2ccc(C3CC3)o2)=O)CC(CNC(C2(C)CC2(F)Cl)=O)O1 11625,C(CN(C)N1CCC(CCN2CCCC2)CC1)c1ccc(OC)cc1 11626,c1(C(N2CCC(C)(C(N3CCC(CF)CC3)=O)C2)=O)ccc(Br)cc1S(C)(=O)=O 11627,N1(C(c2cc(C(C)(C)C)no2)=O)C2CCC1C(NC(c1ccc[nH]1)=O)C2 11628,c1(CSCC(=O)NCC(C)CNC(=O)C(C)O)ccc(Cl)cc1Cl 11629,c1(CSCC(=O)N(C(C)CNC(C2CCO2)=O)C)ccc(Cl)s1 11630,O=C1Nc2ccccc2CC1CC(N1CC2CCCC2C12CC2)=O 11631,C(=O)(C(F)C(F)(F)F)NCC(C)N(C(=O)COC1(C)CCCC1)CC 11632,CC(CC(=O)N1C2CCC1(CNC(c1cc(CO)on1)=O)CC2)C(C)(C)C 11633,C(=O)(CCCCCn1cnnn1)NC(C)(C)CCCNC(=O)CCC1CC1(C)C 11634,c1(C(N2C(C(C)NC(c3cn(CC=C)nc3)=O)CCC2)=O)cc(Cl)ccc1OC 11635,C(=O)(CC1=CCN(C(C2CC2C2CCCC2)=O)CC1)NC(CC=C)C(=O)OCC 11636,CCCCC(O)CC(=O)NCC1CN(C(=O)CNC(N)=O)CCCO1 11637,c1(C(=O)NC23CCN(C(c4c(OC)n[nH]c4)=O)CC2C3)cnc2cc(C)nn2c1 11638,c1(C(=O)NC2CCCC(NC(C(C)(C)O)=O)C2)cnc(O)c2cnccc12 11639,CC12CC(C(=O)NC3CN(C(c4ccc5cnnn5c4)=O)CC3F)(C1)C(C)(C)O2 11640,CCC(O)C(F)(F)C(=O)N(CC(C)(C)Nc1ncnc2[nH]ccc12)C 11641,C(=O)(C1CCc2c(Cl)cccc21)NC1CC2(C(NC(c3cc(=N)[nH]cc3)=O)C2)C1 11642,c1(NC(=O)NCC2(NC(Cc3c(C)cc(C)s3)=O)CC2)cc2c(Cl)cccn2n1 11643,CCC(C(=O)NC(=O)CN1CCC(C)C(CC23CC(CO2)C3)C1C)C(C)(C)CC 11644,c1(OC)cccc(F)c1C(=O)NCCNC(c1ccc(-n2cnnn2)cc1)=O 11645,N1(c2nnc(CC)n2CCC(C)F)CCC(C2CCCCC2)C1 11646,C1(CC)CCC(C)N1C(=O)NC1CN(c2ccc(C(=O)OC)cc2)C1 11647,N1(C(c2c(C)coc2)=O)CC(NC(=O)C(F)(F)c2ccccc2)C(O)C1 11648,N1(C(=O)Nc2c(C)ncc(C)c2)CCC2(CC1)OC(C)(C)NC2=O 11649,C(=O)(CC(C)C(F)(F)F)N1CCC(N(C(=O)Cc2ncsc2Cl)CCC)CC1 11650,c1(C(=O)NC(CC(C)Nc2ncnc(Cl)c2F)C)cc2ccoc2cc1F 11651,C(N=c1cc[nH]c(=NCCCC2CCOC2)[nH]1)c1cnc(C)s1 11652,c1(OC)cc(C)cc(C(=O)NCCOCCNC(C2(S(N)(=O)=O)CCCC2)=O)c1O 11653,C(=O)(C1=C(Cl)CCCC1)NC(C(C)(C)C)C(=O)NCC1CC1C(N)=O 11654,Cc1nc(C)c(C(N2CCN(C3CCCN(C(=O)C=CC(N)=O)C3)CC2)=O)[nH]1 11655,C1(NC(C(CO)OC)=O)CCOC(CNC(c2ccc(C(F)F)cc2)=O)C1 11656,C(CC1=CCN(C(=O)CC2CCCCC23CC3)CC1)NC(=O)CCc1cscn1 11657,N1(C(CC2CC(C)(C)OC2)=O)CC2(CCN(C(c3cc(S(N)(=O)=O)cs3)=O)C2)C1 11658,N1(c2cc(N3CC(C(=C)C)OCC3)ncn2)C2CCC1CC(=O)NC2 11659,N1(C(c2cnn(C)c2C(C)(F)F)=O)CC2CN(C(=O)Cn3ccnn3)CC2C1 11660,Cc1sc(Cl)c(C(N2CCN(C)C(CNC(=O)Cc3nc[nH]n3)C2)=O)c1C 11661,CCC(C)(C(=O)NCCCCCNC(=O)C(CC#N)c1ccccc1)OC 11662,N(C1CCNc2ccccc21)C(=O)CC1CCc2ccccc2C1 11663,c1(CC(=O)NC2(CO)CCN(C(C=C3CCC(C)C3)=O)C2)cccc(Cl)c1F 11664,Cc1ccc(=N)[nH]c1C(=O)NCC(CO)NC(=O)CCn1cncn1 11665,C(CC(=O)NC(C)C(=O)OC(C)C)(CC(C)C)NC(CC1ON=C(CC)C1)=O 11666,C(=O)(CC(F)(F)C(C)C)NCC(CNC(C(COCC)C)=O)CO 11667,CP(C)(=O)c1cc(F)ccc1NCC1(Cl)CC1(F)F 11668,c1(C(N(CCCN(C(CC2(COC)CCCC2)=O)C)C)=O)ccc(C)n(C)c1=O 11669,C(CCN=C(NC1CSC1(C)C)N1CCC(CC(C)C)CC1)SC 11670,C(=O)(C(C)C(=O)N1CCC(n2cc(-c3c(C)noc3C)nn2)C1)OC 11671,CC(C)C(C(=O)N(CC(O)CN(C(=O)C(O)Cc1ccccc1)C)C)NC(N)=O 11672,C1(C(=O)NCCNC(c2cc(O)nc(O)n2)=O)CCc2nnc(O)n2C1 11673,c1(-c2nnn(C(C(C)C)Cc3nn[nH]n3)n2)ccc(Br)cc1 11674,C1(C(N2CCCC(COC)C2)=O)CC2(CC(NC(=O)Cc3ccc(F)cc3)C2)C1 11675,N1(C(c2cc(C)ns2)=O)CC2CC(NC(=O)C(C(C)C)n3cnnn3)CC(C2)C1 11676,c1(CC)cccc(CNC(=O)NC(c2cc(Br)ncc2F)C)c1C 11677,N1(C(c2ccc(C(=O)OC)s2)=O)CCC(NC(C2CCCC(F)C2)=O)C(F)C1 11678,N1(CCNC(C(C)(C)OC(C)C)=O)CCCN(C(=O)CC2CNC(=O)O2)CC1 11679,c12ccc(c(F)c1)OC(=O)CN2.c1(C(C)C)ccc(C(C)(C)OC(=N)O)cc1 11680,C1(CNC(CC2(CNC(=O)C=C3CCCCC3)CC2)=O)CC12CCOCC2 11681,c1(C(=O)NC(c2cn(C)nn2)C(=O)N(CC(F)Br)C)ncc(F)cn1 11682,N#Cc1ccc(F)c(CNC(=NCCCF)NCc2cnccn2)c1 11683,CCC(C(=O)NC1(CO)CN(C(C2CC2c2ccncc2)=O)C1)C(C)O 11684,c1(OC)ccc2c(c1C(=O)NC1CN(C(=O)CC=C(C)C)CC(C)(C)C1)CCC2 11685,C(=O)(C(O)CC(=O)OC(C)(C)C)NCC(CN(C(CC(=C)C)=O)C)O 11686,C(C(C(=O)N1CC(NC(=O)C=CCN2CCCC2)C1)N(C)C)N(C)C 11687,C1(Cc2cn(C3(C(C)(C)C)CC3)nn2)COCCN1C(=O)COC1CCCCC1 11688,C(CC(C)P(C)(C)=O)NC(c1n(CCOCC)nnn1)C1(C(F)(F)F)CCCC1 11689,C=CCC(C(=C)C)C(=O)NC1COCCN(C(c2cc(F)c(Br)c(F)c2)=O)C1 11690,C=CC(C)CC(=O)N1CCCC1C1(NC(c2csc(C(C)(C)C)c2)=O)CC1 11691,C#CCC(C)(C(=O)NC1CCCCC1(C)O)NC(=O)CCOC1COC1 11692,c1(C(=O)NC(C(C)NC(c2cc(CCC)[nH]n2)=O)(C)C)c[nH]c2cc(F)ccc12 11693,N1(C(c2cc(C)nn2C(C)(C)C)=O)CC2CCN(C(=O)CSc3cccs3)C2C1 11694,N1(C(c2cc(C)c(F)cn2)=O)CC(C(=O)NC(C2(O)CCC2)(C)C)CCC1(C)C 11695,C=CCCC(CO)NC(=O)CCCN(C(=O)CC(C)SC)C 11696,c1(-c2ccc(CC)s2)ccc(CNC(C2(CC)CCOCC2)=O)cc1 11697,c1(C(=O)NCC2CCC(NC(=O)Cn3cccn3)CC2)nsc2ccccc12 11698,Cc1ccccc1C(=O)NC1(CF)CCN(C(=O)Cc2cccs2)C1 11699,C1(O)(C(N(CCCN(C(C2CC(=C)C2)=O)C)C)=O)CCCC(C)(C)CC1 11700,N1(C(c2c(CC)noc2)=O)CC2(CCCC2NC(=O)C(c2ccccc2)C)C1 11701,CCCC(CC(=O)NCc1cccs1)NC(c1c[nH]c(=O)cn1)=O 11702,c1(C(=O)NCCCC2OCCN(C(C(CC)C)=O)C2)coc2c1COC2 11703,C=CCCC(C(=O)NC1(C)CC2CCC1C2)NC(=O)C(C)C(F)F 11704,Cc1n[nH]c(C)c1CC(N1CC2C(NC(c3ccncc3O)=O)C2C1)=O 11705,Cc1cc(F)ccc1C(c1ccccc1)NC1(C)CCOC1=O 11706,CN=c1nc(C(=O)NC2CCN(C(=O)CCC(C)(C)OC)C(C)C2)cc(C)[nH]1 11707,Cc1ccn2nc(C(=O)OC3CCN(N4CCN(C)CC4)CC3)nc2n1 11708,C(C(=O)N(C)CCOCCN(C)C(c1cccc(C(F)(F)F)c1)=O)(C(C)C)SC 11709,N1(C(CC2(OCC)CCC2)=O)CC(C(=O)NCCN(S(C)(=O)=O)C2CC2)C(O)C1 11710,C=CCC(CNC(c1cnc[nH]1)=O)NC(=O)CC1COCC1O 11711,N1(C(Cc2ccc(C)cc2C)=O)CC2CC(C)N(C(=O)C3=CCCC3C)C2C1 11712,C1(C(N2C(CC(=O)NCCC(C)OC)CCCC2)=O)CC(C)(C)CN1C 11713,C1(NC(Cc2cn(C(C)(C)C)nc2)=O)CC(NC(=O)C2=CCC2)C(O)C1 11714,C1(C(=O)NCC(C2CCCCC2)C)CCN(C(=O)CCC2CC2(C)C)C1 11715,Cc1ccc(OCCC(=O)NCCCCN(C)C(C2CCCS2(=O)=O)=O)cc1C 11716,CN1CCOC2CN(C(C3CC4CN(C(C5(C)COCCO5)=O)CC4C3)=O)CC12 11717,c1(OCC=C(C)C)ccc(CNC(=O)Nc2n[nH]c(=N)o2)cc1 11718,CCC(C)(C#N)C(=O)NCC#CCNC(=O)CNC(=O)C(F)(F)F 11719,CC(CC(=O)NCCCC1CCCN1C(=O)C=CS(C)(=O)=O)C(F)(F)F 11720,c1(C(C)F)ccc(C(=O)NCCC(C)NC(=O)CC=CCc2ccccc2)cc1 11721,C1(F)(C(=O)NC(CC(=O)NC)C)CCN(C(c2cscn2)=O)C1 11722,c1(CC)nn(C)c(C(=O)NC2CCN(C(c3cnc(O)n3C)=O)CC2O)c1Cl 11723,C(=O)(C1CNC(=O)c2ccccc21)N(C)CCOCc1ccc(F)c2cccnc12 11724,N1(C(c2c(CC)cncc2)=O)CCCC(NC(=O)C(C)CO)CCC1 11725,N1(C(c2nocc2C)C(=O)NCC(=C)C)CCC2(CCc3ccccc32)C1 11726,CCS(=O)c1ccccc1CC(=O)NCC(OC)OC 11727,C1(C2N(C(c3c(C)cc[nH]3)=O)CCC2)CCN(C(C2CN(S(C)(=O)=O)C2)=O)CC1 11728,C1(C(N)=O)(C(c2ccccc2)NC(C(C)SC(C)C)=O)CN(C(C2CC23CC3)=O)C1 11729,c1(OC)cccc(CNC(=O)C(c2n[nH]cc2C)N(C)Cc2c(Br)cnn2C)c1 11730,N1(C(Cn2c(C)cc(C)n2)=O)CCC2C(C1)CN2C(C12CC(C)C1C2)=O 11731,N1(C(C(CNC(CN(CCOC)C)=O)N(C)C)=O)CCCC2OCCC2C1 11732,c1(CC(=O)N(CC2C(CNC(C(C)S(N)(=O)=O)=O)C2)CC)ccc2[nH]ccc2c1 11733,N1(C(C)=O)c2ccc(Cl)cc2CCC1CO.c12ccc(c(O)c1)C(=O)NNC(=O)C2 11734,N1(C(C2CC(CCNC(C3CC4(CCC4O)C3)=O)C2)=O)CCOCC2(CC2)C1 11735,c1(SC)c(C(N2CCC(NC(C3CCC(C)(C)O3)=O)C2C)=O)cnn1C 11736,c1(CNC(C(C2(O)CCC2)NC(c2ccc(CO)s2)=O)=O)ccc(O)nc1 11737,CC1CC(O)CCN(C(=O)C(C)N(C(c2cccc[n+]2[O-])=O)C2CC2)C1 11738,C12(C(N(CC(C)NC(C3(CCC=C)CC3)=O)C)=O)C3CCC(CC13)C2(F)F 11739,C1(NC(Cc2nc(C)sc2)=O)C2CC1N(C(=O)NC1CC1c1ccccc1)C2C 11740,C1(C(=O)NCC(CNC(=O)C=Cc2cnc[nH]2)F)CC2(C1)CC1(CC1)C2 11741,C1(C(N(C2(C(=O)NCc3nc(CC)[nH]n3)CC2)C)=O)CCC(C2CC2)C1 11742,c1(NC(c2n(CC)nnn2)C23CCCC2C3)ccc(OC(C)C)cc1 11743,CC1(C)CC(NC(c2cccc(CC(N)=O)c2)=O)CN1C(=O)CCN1CCC1 11744,C(=O)(C(C)CC(C)(F)F)NC(CC(C)C)(C)CNC(=O)C(F)(F)c1cscn1 11745,CC1CCOC1CNC(c1sccc1CNC(=O)CC1COC(=O)C1)=O 11746,c1(CC(=O)NC2C3(NC(c4cc(C)ns4)=O)CCC(C2)C3)ccc2sccc2c1 11747,C(=O)(CCCCCO)NCC12N(C(C3C(OC)CCC3)=O)CC(C1)C2 11748,c1(C(N2C(C)C(C)N(C(c3ccc(Cl)cn3)=O)CC2)=O)ccc2nn[nH]c2c1O 11749,C1(C(=O)Nc2c(C(=O)OC)scc2)CCCC(NC(=O)NC(C)(C)C)C1 11750,c1(C(=O)OC)cc(NCC(O)COCCN)c(F)cc1F 11751,c1(-c2cn(CC(C)NC(C3CC(C)OC3=O)=O)nn2)ccc(N)c(Cl)c1 11752,C(CS(=O)(=O)CC(=O)N1CCC(C)N(C(c2n[nH]c(C)c2C)=O)CC1)OC 11753,c1(CNC(C=CCN(C)CC)=O)cc(C(=O)NCC(N2CCOCC2)C)n[nH]1 11754,C1(C2CCC2)(C(=O)NCC(CN(C)C(c2ccn(C3CC3(F)F)n2)=O)O)CCC1 11755,C(CCCCC(=O)N1CCCC1)NC(CN(C(C(C)c1cccs1)=O)C)=O 11756,N1(C(C=CC(c2cccnc2)C)=O)CC2C(CNC(C3CN(C)CCO3)=O)C2C1 11757,N1(C(C(CC)OC)=O)CCCCC1CCCNC(C1(OC)CCOCC1)=O 11758,C(=O)(C(C(C)C)NC(c1cc[nH]n1)=O)Nc1c(C)scc1 11759,C=C=CC(C)C(=O)N(C)CCC1CCCCN1C(c1n[nH]cc1Br)=O 11760,c1(C(N2C(CNC(C(CCSC)O)=O)CC(O)C2)=O)c[nH]c2cccnc2c1=O 11761,N1(C(c2cc(C)ncn2)C(=O)NC2CCCC2)CC(CO)C2(CCC2)C1 11762,Cc1ccc2cc(C(=O)NC(C)Cc3cc(Br)ccc3F)cnc2c1 11763,CC(C)(C)CN(CCO)C(C1(CNC(=O)CC2CC=CC2)CC1)=O 11764,C(=O)(CCC(O)C(C)(C)C)N1CCC(CN(C)C(c2cn(CCO)nn2)=O)CC1 11765,N1(C(COCCC#C)=O)CCN(C(c2nnc(C)cc2O)=O)C2CCCCC2C1 11766,c1(CC)nc(=N)[nH]cc1C(N1CCCCCC1CNC(C1CNC(=O)N1C)=O)=O 11767,N1(C(CCC2C(C)=NNC2=O)=O)CCCC(F)(CNC(=O)CC2CC(CF)C2)C1 11768,c1(CC(N2CC(NC(C3C(C(C)C)CCO3)=O)C2)=O)cc2ccccc2cc1O 11769,CC(C)CCCC(C)C(=O)N1CCC(CC(=O)NCCC2(CO)CC2)C1 11770,N1(C(CCSCC)=O)CCC(NC(C23CCC(CC2)CO3)=O)C(F)C1 11771,C1(CNC(c2c(CC)c[nH]c2)=O)CCN(C(c2n[nH]c(C)c2C)=O)C1(C)C 11772,C(c1ccncc1)=C(C)C(=O)N(C1CCCN(C(C2C(C)C2(F)F)=O)C1)C 11773,c1(CC)cccc(S(=O)(=O)N2CCN(C(c3cc(C)c(Br)s3)=O)C(CC#N)C2)c1 11774,c1(C(=O)NCC2=CCN(C(C3CC3F)=O)CC2)cc(F)cc2nc[nH]c12 11775,c1(C(N(C2CCN(C(=O)C(C)C(C)C)C2)CC)=O)ncnc(C)c1C 11776,C12(NC(=O)COc3ccsn3)CCCC1CN(C(=O)CC1COC(=O)C1)C2 11777,C1(C(=O)N(C)C)CCN(CCNC2CC(NC(CCSC)=O)CC2O)CC1 11778,c1(C(=O)NCC(CC)NC(C2C(C=C)C2)=O)cccc(CS(C)=O)c1 11779,C1(C(=O)N(C)CC2(CNC(c3ccc[n+]([O-])c3)=O)CC2)(OC)CCC(C)C1 11780,C1(C(=O)NC2CC(CNC(c3c(C)ncs3)=O)CC2O)CC12CCS(=O)(=O)CC2 11781,CC(C)CC(CO)NC(C1C(CO)CCN1C(=O)CC1(CSC2CC2)CC1)=O 11782,O(NC(=O)C(COCC)NC(=O)CCC1CCOCC1)CC(CC)C 11783,c1(C(=O)NC23CC(NC(c4cccnn4)=O)(C2)C3)ccc(=O)n2c1COCC2 11784,N1(C(CCN(C)C)=O)CC(C(=O)N(C2CCSC2)C)C(F)(F)C1 11785,Cc1ccc(C(=O)NCC(C)CC(=O)NC(c2ncccc2F)C)cc1O 11786,C(CC(=O)N1CCC(CNC(c2nc(Cl)c(Cl)s2)=O)C1)(C(F)(F)F)OC 11787,CC(C(O)C(F)F)NC(C1(N(C(=O)CCOC2CCCC2)C2CC2)CCCC1)=O 11788,c1(OC(CNc2cc(C)c(Cl)cc2)=O)ccc(S(=O)(=O)Nc2conc2C)cc1 11789,N1(C(CC(C)(C)OC)=O)CC2(CCC(CNC(=O)Cc3coc(C(F)F)n3)O2)C1 11790,C1(NC(C=CCC)=O)CN(C(c2c(C)ccn2C)=O)CC1O 11791,N1(C(C2C(C(=O)OC)CCCC2)=O)CC2(CCN2C(c2cnn(C3CC3)c2)=O)C1 11792,N1(C(C2N(C(C)=O)CCOC2)=O)CC2(CCC(NC(c3cc(C)cs3)=O)CC2)C1 11793,C1(NC(C(CO)NC(C(C)C)=O)=O)CCCN(Cc2ccccc2)C1 11794,CC1CN(CC(Cl)=CCl)CCC1N(C)C.C12(CCC1)C(=O)N2 11795,c1(C(=O)NCC2CCCN(c3nccc(CO)n3)C2)cnc(O)c(C(F)(F)F)c1 11796,C1(NC(COCCCC)=O)CCN(CCNC(=O)CN2CC3CC3C2)CC1 11797,C(=O)(C1=CCN(C(c2cc[nH]n2)=O)C1)NC(c1ncc[nH]1)(C)C 11798,C(=O)(CC(C)(C)N(C)C(C1(C(C)(F)F)CC1)=O)N(CC(COC)O)C 11799,Nc1cc(NC(=O)NC(CO)CCc2ccccc2)on1 11800,c1(CNC(CSC)=O)cc2cnccc2o1.c12ccc(cc1)[nH]c2=O 11801,c1(CC)nn(C)c(C(N2CCSCC2C(N2CCOC3CC23)=O)=O)c1Cl 11802,C(=O)(CCC(=O)OC(C)(C)C)NCC(CN(C(=O)CN1CC(=O)NC1=O)C)O 11803,C(=O)(C1=CCN(C(C2(F)CCCC2)=O)C1)N(c1cnc(F)nc1)C 11804,N1(C(c2ccc3c(n2)NCC3)=O)CCCC2CN(C(C3(F)CCC3)=O)CCC12 11805,N1(C(C(C)OC)=O)CC(CNC(=O)C(c2ccc(C)cc2)C)C2(CCC2)C1 11806,Cc1cc(C(N2CC(NC(=O)C(F)F)C(F)C2)=O)c(C)n1-c1ccc(Br)cc1 11807,C1(N(C(C(C=C)O)=O)C)CCC(CNC(=O)C(COC)N(C)C)CC1 11808,C(CCC(F)(F)F)(c1cccnc1)C(N1CCC1Cn1cc(C2CC2)nn1)=O 11809,CCC(O)CC(=O)NC(CC1CC1)C(=O)N(C)CC1CCCC2CC12 11810,CCC(C)(O)C(=O)NCC1(F)CCC(CNC(=O)C=C(C)I)C1 11811,c1(C(N2CC(CC(=O)N(CCCCCC)CCO)(OC)C2)=O)ncn2c1CCC2 11812,CC1Cn2nccc2CN1C(=O)C1=C(F)CN(C(=O)CCc2ccnn2C)CC1 11813,CCC(CC(=O)N(C1CCCCC1CC)C)N(C(=O)CN(C1CCC1)C)C 11814,C1(NC(C=CC(C)(C)C)=O)CCN(C(=O)CC2CC2C2CC2)C1c1ccccc1 11815,c1(NC(N2C(CCNC(C3C4CCOCC34)=O)CCC2)=O)cnccc1CO 11816,c1(CC)cnc(C)nc1N1CCC(C(F)(F)F)(Nc2cnc(OC)cn2)C1 11817,N1(C(C(C)(C)OC)=O)CC2(CCCN(C(=O)CC3CCCC(=O)C3)C2)C1 11818,c1(C(N2C(C)CC(NC(c3c(C)cc(C)nc3)=O)C2)=O)ccc2nc(S)[nH]c2c1 11819,c1(C(=O)C(C)=O)cccc(C(N2CCC(C)C2)=O)c1.N1(C)CCN(C(C)C(C)(C)O)CC1.O 11820,c1(CN(CC)CC)cc(F)ccc1C(=O)NC1(C2CC2)CCOC1 11821,c1(C(=O)NC(CN(C(C2(C)CCC(F)(F)C2)=O)CC)C)cnc(C(C)C)nc1C 11822,CC1CCN(C(c2n[nH]cc2Cl)=O)C(CNC(c2cc(-c3ccco3)on2)=O)C1 11823,N1(C(c2c(C)nc(Cl)s2)=O)CCc2sc(C(=O)NCC3COC3)cc2C1 11824,N1(CC)CCC(C(=O)NC2CCCCC2CNC(c2cnsc2C)=O)CC1 11825,C(CN=C(NC(C)COC)NC1CC2(CC2)C1)OC 11826,C1(C(N(CC2=CCSC2)C)=O)C2CCC(C2)N1C(C1(C)CCC1)=O 11827,N1(C(c2c(Br)cn(CC)n2)=O)CCC2C(CCCN2C(=O)CC23CC(C2)C3)C1 11828,C(CNC(=O)CC(C)(C)C)(C(C)C(C)C)NC(c1c(COC)cccc1)=O 11829,c1(C(N2CCCC(NC(C3CCC4CC3CO4)=O)C2)=O)nc2c(s1)COCC2 11830,C1(NC(C(C)(C)N2CCC2)=O)CC2(C1)CC2C(N1CCC(O)(C(F)(F)F)C1)=O 11831,c1(C(N2CC(n3cc(CNC(CC)=O)nn3)C2)=O)cc(Cl)cn1C 11832,C(C(=O)NC(C)CC)(C(C)CC1CC(F)(F)C1)N(C1CCCC1)CCC 11833,c1(C(=O)NC2C(NC(C(C)CN(C)C)=O)CCCC2)ccc2c(O)ncnc2c1 11834,CC1(C(=O)NCC2CC(O)(CNC(=O)CNC(C3CCC3)=O)C2)CCOCC1 11835,C#Cc1cncc(C(=O)NCCC(C)(C)NC(c2cncn(C)c2=O)=O)c1 11836,Cc1cc(NC2(CNC(=O)CCCC3CCC3)CCOCC2)nc(S(C)(=O)=O)n1 11837,Cc1ncsc1CNC(=O)C(n1cc(-c2ccsc2C(=O)O)nn1)C 11838,c1(C(=O)NC2CCCC(NC(c3ncc(C)c(Cl)c3)=O)C2)cc([N+](=O)[O-])cn1C 11839,n1(CC(N2CC(C(C)NC(Cc3c(C)n[nH]c3)=O)C2)=O)nc(C)n(C)c1=O 11840,C(=O)(CCCCCC(C)(C)C)NCCCN(C(C)C)C(C1CC12CCOCC2)=O 11841,c1(NC(c2cncnc2)COC)cnc(COC)s1 11842,C1(NC(CSCC(=O)OCC(C)C)=O)CN(C(=O)CCOC(C)C)CCC1C 11843,N1(C(c2c(C)nc[nH]2)=O)CC2CC(NC(c3cc(N)ccn3)=O)C(C2)C1 11844,C1(C(=O)NC2(CNC(CCC(C)C)=O)CC2)Cc2ccccc2N1C(C)=O 11845,c1(CNC(=O)NC2(C(=O)O)C(C)C2)cc(Cl)cc(Br)c1 11846,N1(C(C2(CCNC(CCC(C)OC)=O)CCCC2)=O)CCSCC(C)C1 11847,N1(C(c2cc(C)nc(O)c2)=O)CC(CNC(c2nccnc2Cl)=O)OC(C)(C)C1 11848,N1(C(c2c(CC)ocn2)=O)CCCC2(C1)CN(C(c1c(C)noc1C(C)C)=O)C2 11849,Cc1nc(C(=O)NCC2C=CC(NC(=O)C(O)CC3CCOCC3)C2)sc1C 11850,N1(CCOC)CCOC2(CCN(C(C3CCC4CCCCN34)=O)CC2)C1 11851,Cc1ccccc1C(=O)NCC(N1CCOCC1CC(=O)NC1COC(=O)C1)=O 11852,N1(C(C(C(C)C)CNC(C2CCN2C)=O)=O)CC2(C1)CC(C)(O)C2 11853,c1(CC)cccc(C(=O)N(CC(C)N(C)C(c2ccc(Br)cc2)=O)C)c1 11854,CCCC(C)CCNC(c1nnnn1CCCF)c1cn[nH]c1 11855,N1(C(C(c2cccnc2)NC(C(C)n2cccn2)=O)=O)CC(CO)C(C)C1 11856,Cc1c(F)cc(C(N2CC(NC(c3cccnc3F)=O)C(C)C2)=O)cc1Br 11857,N1(C(c2cc(CC)[nH]n2)=O)CCC(C2CCN(C(=O)CCCC(=O)N(C)C)C2)C1 11858,Cc1ccc(=O)n(CC(N2CC(NC(c3cc(C(C)(C)C)n[nH]3)=O)CC2C)=O)n1 11859,N1(C(C(CC=CC)CC)=O)CC(C2CCN(C(=O)CCNC(N)=O)CC2)C1 11860,CCCCCCC(C)C(=O)NCC1CC2CN(C(=O)C(F)(F)C(F)F)CC12 11861,c1(CN2C(CCOC)CCC2)ncc(Br)cc1Br 11862,N1(C(c2cccc(COC)c2)=O)CC2CCCC2(Nc2nc(C)cc(C)n2)C1 11863,C#Cc1cccc(C(N2CCCC2(C)C(=O)NC2CC=CC2)=O)c1 11864,C(=O)(C1=CC2CCCC12)NC1(CNC(c2cc(C)cc(OC)c2O)=O)CCC1 11865,CC(C)CC(=O)C(=O)NCC(C(N1CC(CO)CC(C)C1)=O)N(C)C 11866,C(=O)(CS(=O)(=O)C(C)(C)C)N1CC(C(N)=O)(CNC(Cc2c(C)nc(C)s2)=O)C1 11867,Cc1c(C(=O)NCCn2cc(C(=O)NC(c3ncnn3C)C)nn2)ccn1C 11868,C1(C(N(CCN(C(CC2C(C)=NNC2=O)=O)C)C)=O)SC2C=CC1CC2 11869,n1(CC)nc(C(N2CC3CC3(NC(C3CCC(C(F)(F)F)CC3)=O)C2)=O)cc1O 11870,CCC(c1cccc(Cl)c1)=CC(=O)NC1CCC(CNC(C2CNC(=O)N2)=O)C1 11871,C(=O)(C(CC(C)(C)C)NC(C1CC(=O)CCO1)=O)NC1CCC(C)(OC)CC1 11872,C(CN=c1ccc([N+](=O)[O-])c[nH]1)NCOCCNC(c1scnc1Cl)=O 11873,C1(NC(COCCCOC)=O)CCCC2CN(C(=O)C(C)CS(C)(=O)=O)CC12 11874,N1(C(CC(C)O)=O)CCCC2(CCCN(Cc3ccc(F)c(O)c3F)C2)C1 11875,C1(NC(c2c(CC)nn[nH]2)=O)CC=CCC1C(=O)NC(C(C)C)C1CC1 11876,C1(C(N2CCC(N(CC#C)C(C3COCCO3)=O)C2)=O)CCCCC1(C)C 11877,c1(CN(c2n(C(C(CC)C)C)nnn2)C)ccc(Cl)cc1 11878,C#CC(C)(C)C(=O)NC(C1CN(C(=O)C=CCN(CC(F)(F)F)C)C1)C 11879,c1(C(C)(C)C)c[nH]c(C(=O)NC(CNC(=O)CCC2CCCCO2)CO)c1 11880,c1(C(=O)NCC2CC2CNC(c2cnsn2)=O)cc(=O)n(-c2ccccc2)[nH]1 11881,N1(C(CCn2c(=O)ccc(C)n2)=O)CC2OCCN(C(=O)Cc3ccsn3)C2C1 11882,Cc1cc(CN2CCC(C)(NC(c3cc(C)n(C)n3)=O)C2)c(C)s1 11883,N1(C(C(C)NC(CC)=O)=O)C2CCC1CN(C(c1c(C)nc(C)n1O)=O)C2 11884,Cn1cc(Br)cc1C(=O)NCC1CC1NC(c1cncnc1C1CC1)=O 11885,c1(C(=O)NC2CC(CNC(C(C)O)=O)C2)ncoc1C1CC1 11886,c1(C(=O)NCCN(c2[nH]cnc3nc(Cl)cc2-3)CCC)cc(F)cc2nn[nH]c12 11887,C1(CC(=O)NC(C(=O)OCCC)C)CC(C)N(C(=O)CC2CCCC(=O)C2)C1 11888,Cc1cc(F)cnc1C(N1CCCC1CCNC(C1(C(F)(F)F)CCC1)=O)=O 11889,N1(CCNC(C2C=CCC2)=O)CCCN(C(=O)Cc2csc(C3CC3)n2)CC1 11890,N1(C(=O)C2=CCCO2)CC2CCCN(C(C3C=CCCC3)=O)C2C1 11891,N1(C(c2c(NC(c3c(C)nns3)=O)cccn2)=O)CCCC(S(C)(=O)=O)C1 11892,c1(CCC(N2CCCC(n3cc(COC(=N)O)nn3)C2)=O)ncc(Br)cn1 11893,C(=O)(C1=CCCC1C)NCc1cc(C(=O)NCC(C)OCC=C)on1 11894,N1(C(C(CCCC)(C)F)=O)CCC2(CCN(C(c3c(C#N)cnn3C)=O)CC2)C1 11895,c1(C(=O)NCCC2N(C(C=C(C)C(C)C)=O)CCCC2)cccc(Br)c1N 11896,C1(N(C(CC2(COC)CC2)=O)C)CCCN(C(c2c(C)ccn2C)=O)C1 11897,N1(C(C(=O)N(C)C)=O)CCC2CCN(C(=O)Cc3coc4ccccc34)CC12 11898,CCC(C)(CNC(c1ccc(F)s1)=O)NC(=O)CN(c1ncccn1)C 11899,N1(C(C2CCN(C(C)=O)CC2)=O)Cc2[nH][nH]c(=NC(=O)C3CC3F)c2C1 11900,C(=O)(C(CC(F)F)c1ccccc1)NCC(CC=C)NC(=O)OC(C)(C)C 11901,C1(C(N2C(CC)C(NC(=O)CN(CC)CC)CC2)=O)CC2(CC(OC)C2)C1 11902,C(=O)(C1=C(F)CN(C(C2CC(n3ccnn3)C2)=O)CC1)N(C1CC2CC2C1)C 11903,N1(C(C2C(C)N(C)CC2)=O)CC2(CCNC(=O)CCC(N)=O)CCC1C2 11904,CC(Cc1ccc(Cl)cc1)CC(=O)NCC1CCN1C(=O)Cc1cnccn1 11905,Cc1ccc(NC(=O)CSCC(N2CCC3C(Br)C3C2)=O)c2ccccc12 11906,N1(C(C(CCC(C)(C)C)F)=O)CCCCC(C2CN(C(C3CCC(=O)N3)=O)C2)C1 11907,c1(NC(N2CC(C)(CC(=O)NC3CNC(=O)C3)C2)=O)ccc(Cl)cc1 11908,N1(C(=O)C(C2CCOCC2)O)CC2CCCC2(Nc2cc(Cl)ncn2)C1 11909,C1(F)(NC(=O)NC(C(=O)O)C2CCCC2)CN(C(=O)OC(C)(C)C)CC1C1CC1 11910,CC1CCCC(C)N(N(C2CCNCCC2C)c2cnn(-c3ccccc3)c2)C1 11911,C(=O)(CC(=O)N(CC(C)C(=O)NCCCC(=O)NC)C)OCC 11912,C12(CNC(C(C)OCc3ccncc3)=O)CCCCC1N(C(=O)C(C)O)CC2 11913,N1(C(C(CC)C(F)(F)F)=O)CCC(C2CCN(C(=O)CCn3cnnn3)CC2)C1 11914,c1(C(N(C)CCN2CCN(C(=O)CC34CC(C3)C4)CC2)=O)ccc(F)cc1Cl 11915,CC1(C)CC(CNC(=O)C(F)=CC2CC2)CN(C(=O)CN2CC3CC3C2)C1 11916,Cc1ccncc1C(=O)NCc1cn(CCNC(=O)Cc2ccns2)nn1 11917,C=CC(CC)CC(=O)N1CCN(CCCNC(C2(S(C)(=O)=O)CC2)=O)CC1 11918,N(C(=NCCCF)N1CCCC(S(C)(=O)=O)C1)C1(c2c(C)nccn2)CC1 11919,c1(C(=O)NCCCCn2cc(C3CC(F)(F)C3)nn2)cc(Br)cc(I)c1F 11920,C1(CCNC(CC2(C)OCCO2)=O)CCCN(C(c2cnc(Cl)s2)=O)CC1 11921,c1(C(C(=O)NCC2CCC(NC(c3nsnc3O)=O)C2)(F)F)ccc(F)cc1F 11922,C=CCC(CC)C(=O)NC1(C(=O)NOCC(=O)OCC)CCN(C)C1 11923,Cc1cncc(C(N2CC(NC(c3cc(-c4cnn(C)c4)[nH]n3)=O)C(F)C2)=O)n1 11924,c1(C(=O)NC2C(C)CN(C(c3cccn(C)c3=O)=O)C2)cccc2c1CCCC2 11925,c1(C(N2CCCC(CCNC(C(CC)CO)=O)C2)=O)ccc2nonc2c1 11926,C1(CNC(CC(=O)NCC)=O)CCN(C(=O)CN(c2ccnc(Cl)n2)C)CC1 11927,c1(CNC(C2CC2F)=O)ccc(CNC(=O)Cn2cc(CO)nn2)cc1 11928,N1(C(C(C2CCCCC2)NC(C(=O)NC(C)C)=O)=O)CCS(=O)(=O)CC1 11929,C1(C(=O)NCC2CCN(C(C3CCO3)=O)CC2(F)F)CCC2(CCCC2)CC1 11930,N1(C(CCCC#CC)=O)CCC2(CCC2NC(=O)Cc2ccc(C)nc2)CC1 11931,n1(CC(CC)C)c(N(C)Cc2cccc(Cc3ccccc3)c2)nnc1C1CC1 11932,C1(C(N2CC(NC(CSCC#C)=O)(CO)C2)=O)CCN(C)C1C 11933,N1(C(COCCCC#C)=O)CCC(C2N(C(=O)C=CC(C)C)CC2(C)C)CC1 11934,C(=O)(C1=C(C)CCCC1)NCC12N(C(C(CCCC)O)=O)C(CC1)CC2 11935,C(=O)(C(CC)C(C)O)NCCN(C(C=C(CCC)CCC)=O)CCOCCO 11936,c1(CNC(COCC(=C)C)=O)ocnc1C(=O)NC(C)Cc1cccnc1 11937,N1(CCC)CCc2cc(C(C)NC)ccc21.C1(C)CN1C(C)=O 11938,C1(NC(C2N(C)CCC2)=O)CCN(C(c2cc(=N)[nH]cc2Br)=O)C1(C)C 11939,CCCC(C(=O)N1CCC(N(C)C(c2ccc(O)c(F)c2F)=O)CC1)S(N)(=O)=O 11940,CC1OC2CCC1(C(N1CC(NC(c3cc(Cl)cs3)=O)C1)=O)C2 11941,c1(OC)ccc(C(=O)NCC(C(C)(C)C)NC(c2ccsc2)=O)cc1C(F)F 11942,C1(C#N)(C(=O)NCC(C2CCCC2)NC(C(C2CCOCC2)C)=O)CC=CC1 11943,C(=O)(CCCCCC(C)(C)C)NCC(CNC(CN1CC(CC)C1)=O)O 11944,C(CC(O)C(=O)N1CCC(CCc2cn(Cc3cccnc3)nn2)CC1)N(C)C 11945,C1(C(N2C(C(C)(C)NC(=O)CC3CCCC(O)C3)CCC2)=O)CC(S(C)(=O)=O)C1 11946,C12(NC(=O)NC3CCCC3CNCc3nc(C(F)(F)F)cs3)CCCN(CC1)C2 11947,N1(C(=O)CC2CCCO2)CCN(C(c2cnc(O)o2)=O)C(c2ccccn2)C1 11948,C1(CNC(c2ccc(OCC)cc2)=O)CC2CCC(C1)N2C(=O)C(F)CC 11949,c1(OCC=C)ccc(CCNC2CC(=O)N(c3ccccc3Cl)C2)cc1 11950,C1(C(=O)NC(C2(O)CN(C(Cc3cc(C)[nH]n3)=O)C2)C)CCc2nccn2C1 11951,C#CC(CNC(=O)C(C)N(C(=O)C(CCC)N(C)C)CCC)CC(C)(C)C 11952,C1(CCNC(c2cn(CC=C)nc2)=O)CCCN(C(=O)CCc2nc[nH]n2)CC1 11953,C1(O)(CCNC(C2CCOC2)=O)CCN(C(c2cnn(CC(F)F)n2)=O)C1 11954,c1(OCC)cc(C(=O)NC(C)C=CC(=O)N(CCCOC(C)C)C)[nH]n1 11955,c1(OCC(=O)NCC2(CNC(C3N(N=O)CCC3)=O)CC2)ccccc1[N+](=O)[O-] 11956,c1(N2CC(O)(CCNC(C=COCC)=O)C2)ncc2cccnc2n1 11957,N1(C(C2CCCC(NC(C3CCOC3)=O)C2)=O)CCN2CCCCC1C2 11958,C1(NC(C2ON=C(CC)C2)=O)CC2CCCC(C1)N2C(c1nonc1N)=O 11959,c1(C(N2CCC(CC=C)(NC(C3COC(C)C3)=O)C2)=O)cc([N+](=O)[O-])cnc1O 11960,N1(C(c2c(CC)noc2)=O)CCC2(CC1)CN(C(=O)CSCc1ncc[nH]1)CCO2 11961,N1(C(C(C(CC)(F)F)(C)C)=O)Cc2ccccc2-c2ccccc2C1 11962,C1(C(N2CC(OC)(CNC(C3CCCC3O)=O)C2)=O)C2(CCC2)C12CCC2 11963,c1(CN(C)C(c2ccon2)=O)ccccc1CNC(c1cc(Cl)ns1)=O 11964,N1(C(CCCOC(C)C)=O)CCCC(C(C)NC(=O)CCCCC2CC2)C1 11965,c1(-c2cn(CC(=O)N(CCC)CCN(C)C)nn2)ccc(COC)nc1 11966,c1(COC(c2sc(OC)c(Br)c2)=O)c(F)cc(F)c(O)c1F 11967,c1(C(=O)NC2CCN(C(C3CCN(C4COC4)C3)=O)C2)ccc2c(c1)NCC2 11968,N1(C(CCCCC=C)=O)Cc2ccnn2CC(NC(c2nc(CC)c[nH]2)=O)C1 11969,N(C1CCc2cc(Br)ccc21)C(N1CC(c2ccccn2)C1)=O 11970,Cc1ccc(C)c(C(=O)NC2CCN(C(=O)CSc3ccccn3)CC2F)c1C 11971,c1(C(=O)NC2C(C)CN(c3nc(C#N)ncc3Cl)CC2)ccc2ncccc2c1 11972,c1(OC)ccc2c(C(=O)NC(C3CCCCN3C(c3ccns3)=O)C)n[nH]c2c1 11973,C(CCCCC(=O)NC1C2CCC(F)(F)C12)NC(=O)CC1CCSC1 11974,C1(NC(=O)CC2CCCCCO2)CC2CCC(C1)N2C(C1(CC(F)(F)F)CC1)=O 11975,O(N=C1CCCCCC1)CC(=O)NC1(COC)CN(C(C23CCCC2C3)=O)C1 11976,c1(C(c2nnnn2C)NCC(CCCC)CO)ccc(S(=O)(=O)NC)cc1 11977,CC1(C)CC(C(=O)NC2(c3cc[nH]n3)CC2)(CNC(C2CCC(F)(F)C2)=O)C1 11978,c1(C(N2C(CNC(c3n(CC)ncc3)=O)C(C)CC2)=O)ncc(Cl)cc1Cl 11979,CC1(C(=O)NC2CCC(F)(F)C2O)C2Cc3ccccc3C12 11980,CC1(C)CC(C(N2CC(Cc3ccco3)C2)=O)N(C(=O)CC2CCC=CCC2)C1 11981,C(CCC(=O)NCC1(C(N2CC(CC)C2)=O)CC=CC1)=CCC=C 11982,C1(NC(CN(C(C2CC(C(N)=O)C2)=O)C2CC2)=O)CCn2nnnc2C1 11983,CC(C)CC(F)C(=O)N1CC(CNC(c2csc3nnsc23)=O)C1 11984,c1(C(=O)NC2CCCN(C(C(C)(C)N(C)C)=O)C2)cc2n(n1)CCN(C)C2 11985,c1(SC2C(C(=O)NCC(C3CCCCC3)NC(C)=O)C2)ccccc1 11986,CCCCC(C(=O)NCC1(O)CCN(C(=O)Cc2cnccc2Cl)CC1)C(C)C 11987,C(=O)(C(C)(C)C1=CCN(C(=O)C(C2CC2)C2CC2)C1)NCC(C(CC)C)CO 11988,n1(CC(=O)NCC(C)(CNC(=O)CCOC2CCCC2)OC)nc(C)nc1C 11989,O=C(C1=CC2(CCOC2)C1)NCC1CCN(C(c2cc(=O)cc[nH]2)=O)C12CC2 11990,c1(N(C)Cc2ncccn2)nc(N2CCCC(CC(F)F)C2)nc2c1ncn2C 11991,c1(C2(C)C(NC(=NCC=C)NCCF)C2)ccc(OC)c(OC)c1 11992,O=S(=O)(c1cc(Br)cc(Br)c1)N1CCn2c(C3CC3)nnc2C1 11993,c1(C(=O)NCCC2(O)CN(C(C(CC#C)C)=O)C2)cc(NC(C)=O)cc(Cl)c1 11994,C1(CNC(CC)Cc2ccc(C)cc2)Cc2cccc(C)c2O1 11995,c1(C(=O)NC23CC(NC(c4ccc(C(N)=O)cc4)=O)(C2)C3)cnc2[nH]nnc2c1 11996,c1(OC)cc(C(=O)NC2CC(C(=O)Nc3cnc(C)s3)C2)ccc1O 11997,c1(C(=O)NC(CNC(C2(C#C)CC2)=O)CC(C)C)ccc(Cl)c(CCC)c1 11998,CC1(C)CC2(CC(C(=O)NCC(O)CNC(=O)CP(C)(C)=O)C2)C1 11999,S(=O)(=O)(c1ccc2c(c1)OCO2)N1CC(NC(c2csnn2)=O)C(F)(F)CC1 12000,C1(C(=O)NC2C(C)(C)CC(O)C2)CC2(CCN(C(C3C4(CC4)C34CC4)=O)C2)C1 12001,N1(C(=O)Nc2ccc(N=S(C)(C)=O)cc2)Cc2ccccc2C(C(=O)O)C1 12002,Cc1cc2sc(C(=O)NCC(C(C)C)NC(=O)C(C#N)C(C)C)cc2s1 12003,CC(C)(CNC(=O)CC(C1CCC1)C1CCC1)N=c1[nH]nc(C#N)s1 12004,c1(OC)ccc(O)cc1NC(=O)CCCN(C(=O)C(C)(C)C(C)O)C 12005,CCC(O)(CC)CCNC(C1CC(NC(c2c(C)n[nH]c2C)=O)C(O)C1)=O 12006,c1(C(N2CCC(NC(C(CC=C)C)=O)(CO)C2)=O)cccn2c(CO)nnc12 12007,C1(N(C(CC2(C(=O)OCC)CCC2)=O)C)CCCCC1N(C(=O)C1=NOCC1)C 12008,c1(C(N2CC(CNC(c3nc(C)nn3C)=O)C(C)C2)=O)cc(Cl)cc2c1CCC2 12009,C1(NC(C2CC3CCC2C3)=O)CCCC(CC(N2CCC(F)CC2)=O)C1 12010,CC(C)C(Br)C(=O)c1ccc(C2CCN(C)CC2)s1 12011,C1(c2n(C(CC)C)nnn2)(Nc2cnn(CC(C)C)c2C)CSC(C)(C)C1 12012,N1(C(c2c(N)cncc2)=O)CC2(CCCC2NC(=O)COCCF)C1 12013,C(=O)(C(C)(C)CCC#N)NCCC1N(C(c2scc(OC)c2)=O)CCCC1 12014,C12(NC(C(CC#CC)NC(=O)CC(COC)COC)=O)CCC(CC1)C2(C)C 12015,c1(C(=O)NC(CN(C(c2ccc(OC)c(F)c2)=O)C)C)csc2c1CCC(C)C2 12016,c1(C(COC(c2ccnn2CCN(C)C)=O)=O)cccc(-n2cnnn2)c1 12017,C(CC(C(=O)NCC1CC(NC(=O)CC2C=CCC2)C1)c1ccccc1)=CC 12018,c1(N2CCC(NC(=O)Cc3cccc(Cl)c3)C(O)C2)ncnc2ccc(O)cc12 12019,N1(C(CC2(C)CCC2)=O)CCC(C)(C)C1C(=O)Nc1cccc(CO)c1 12020,c1(C(N2CCC(NC(c3nn(C)c(Cl)c3)=O)C2)=O)c(F)cncc1Cl 12021,C(=O)(C(O)CC(F)(F)F)N1CC(CCCCNC(c2ccc([N+](=O)[O-])o2)=O)C1 12022,c1(C(CNC(C2CN(C)C2)=O)NC(C(C)=C2CCCC2)=O)ccccc1 12023,C(=O)(CCCCCC(C)C)N1CCCC(CCC(N2C(CC)CCC(C)C2)=O)C1 12024,c1(OCC)nc(N2CCCC2CNC(C23CCCC(C2)OC3)=O)ncc1Cl 12025,C1(C(=O)NC2CN(C(c3c(C(C)C)ocn3)=O)CC2C)CCC2(C1)CC2(F)F 12026,CC1(C)CN(C(=O)C(F)F)CCC1NC(=O)CCc1ccc(F)cc1Cl 12027,N1(C(C(C)SC)=O)CCC(C2CCN(C(c3cn(C)nc3C(F)(F)F)=O)CC2)C1 12028,CC1(C)COCC1C(=O)NC1CCC(NC(C2(C(F)F)CCCO2)=O)CC1 12029,c1(C(=O)NC2CC3CN(C(c4ccc(Br)o4)=O)CC23)cccn2cncc12 12030,C(=O)(C1=CCC(C)CC1)N1CCN(C(c2ccc(C)cc2F)=O)C(CF)C1 12031,Cc1cc(C)n(CC(=O)NCc2cc(C(=O)NCC(c3ccnn3C)O)co2)n1 12032,c1(C(N(C)CC2N(C(C(C)NC(N)=O)=O)CCC2)=O)ccc(Cl)c(Br)c1 12033,C(=O)(C(C(C)(C)C)NC(C1CC2(CC2)CN1C)=O)NC(c1ccns1)C 12034,C1(NC(c2c(SC)cccn2)=O)COC2(CCN(C(C3OCCO3)=O)C2)C1 12035,C(=O)(C1=C(F)CN(C(C2COCCO2)=O)CC1)NCC(C(C)O)O 12036,C(N=c1nc2c(ncn2C)c(N2CCC=C(C)C2)[nH]1)c1c(OC)nn(C)c1 12037,C12(C(N(CC#C)C)=O)C(NC(=O)C=C(C3CC3)C3CC3)C3CC1C2C3 12038,CC1C(NC(C2CCN(C3CC3)CC2)=O)CCCN1C(=O)CN1CC2C=CC1C2 12039,C(C(C(=O)N(C1(C2CC2)CC1)C)NC(C1CCC(=O)O1)=O)N(C)C 12040,C1(C#N)(C(N2CCC(CN(C)C(c3ccnc(CO)c3)=O)CC2)=O)CCCC(=O)C1 12041,C1(CC(N)=O)CCN(C(C2CC(n3cnnc3)C2)=O)C2(CC2)C1 12042,Cc1[nH]nc2ncc(C(=O)N(C3CCNCCC3C)c3cnccc3Cl)cc12 12043,C1(C(=O)NC2CCC(NC(CCc3cc(C)on3)=O)C2)CCC2(CCCCC2)C1 12044,c1(SC)cc(C(=O)NCC2(NC(C3C=CC(CO)C3)=O)CCC2)ccc1N 12045,Cc1ccc(F)c(C(N2CC(CNC(=O)C(C3CCOCC3)C)C(O)C2)=O)c1 12046,C(=O)(C#CC1CCOCC1)N1CCC(C(N2CCCC(CC(C)C)C2)=O)C1C 12047,c1(C(=O)NCCCCCN(C(=O)CC2(C)CC2(Cl)Cl)C)cc([N+](=O)[O-])cnc1N 12048,N#Cc1ccc(N2CCCC(NC(=O)NC(c3ccccn3)CCO)C2=O)cc1 12049,N1(C(CC=C)=O)CCCN(C(=O)C(c2ccc(OC)c(F)c2)C)C(CC2CC2)C1 12050,c1(CC)cccc(C(=O)N(C)CC2(NC(c3cc(C4CC4C)on3)=O)CC2)c1F 12051,Cc1cc(C(=O)NCCn2cc(C(=O)NC(C)CS(C)=O)nn2)ccn1 12052,C1(N(C(C(COC)N(C)C)=O)C)CN(C(c2cn(C)nn2)=O)CC1O 12053,C(C(=O)CCC(=O)N=c1ccn(CC(C)C)[nH]1)OCCOC 12054,C#Cc1ccc(C(N2CC3CC3(C(=O)NC(c3nnc(O)n3C)C)C2)=O)cc1 12055,CCC(C)CCCC(=O)N1CC=CC1C(=O)N(C)CC1CN(C)CCO1 12056,c1(OC)ccc(CCC(=O)NCCC(C)NC(C2CC2CC(C)C)=O)cc1C 12057,C1(O)(C(C)NC(=O)CCCOC2CCOCC2)CCN(C(=O)Cn2ccnn2)C1 12058,C1(NC(=O)C(C2(O)CCC2)NC(C2CC(C3CC3)C2)=O)CC2CCC(C1)S2 12059,Cc1cc(=O)n(CCC(=O)NC23CC(NC(=O)CSc4n[nH]c(=N)s4)(C2)C3)cn1 12060,N1(C(CCC=CCC=C)=O)CCOC(CN(C)C(C2CC(F)C(=O)N2)=O)C1 12061,c1(C(=O)NC(C)CNC(c2nscc2Br)=O)ccnc(OCCO)c1 12062,c1(C(C)(C)C)c(C(N2CCC(CNC(=O)COC3CC3)(OC)C2)=O)cccc1F 12063,C1(COC)(NC(=O)CCNC(N)=O)CCN(C(c2cc(F)cc(Cl)c2)=O)CC1 12064,c1(OC)cc(NC(=O)CC(n2nc(C)cc2C)C)cc(OC)c1C(C)C 12065,Cn1cc(C(=O)NCC2(C)CC(NC(c3ocnc3C3CC3)=O)C2)c(=N)[nH]1 12066,N1(C(c2c(CC)cns2)=O)CC(O)CC1C(=O)NC(COC)C(C)C 12067,C1(NC(CCCC)=O)CC2(CCN(C(=O)C(C(C)C)N(CC)CC)CC2)C1 12068,c1(SCCc2nc(C3(C(F)F)CCNC3)on2)ccc(Cl)c(Cl)c1 12069,CCCCCCCCC(=O)NCC(C1CC1)NC(=O)C(CC)C(=O)OCC 12070,N(C(=NCc1ccc(C)cc1)NC1CCOCC1)CC(C1CCOCC1)OC 12071,C1(OC)C(OC)CN(C(=O)C(C)C2CC2)C1CNC(c1nc(Cl)sc1C)=O 12072,C1(CC)COCCC1(c1nnnn1Cc1ccccc1)Nc1ccc(F)c(F)c1 12073,C1(NC(CCC=CC)=O)CC2(CCC(CNC(c3cc(CCC)on3)=O)CC2)C1 12074,Cc1ncccc1C(=O)NC1(CCC(=O)Nc2cncc(C(N)=O)c2)CCCC1 12075,C1(OC)CC(CNC(=O)C=Cc2ccnn2C)N(C(c2cc(C)on2)=O)C1 12076,c1(C(=O)NC(C2CN(C(CC(C)SC)=O)C2)C)ncnc(C)c1C 12077,C(=O)(C(=O)CC(C)C)N1CCC(C(C)NC(C2(OCC)CCC2)=O)CC1 12078,C1(C(N2C(C3(N(C)C(c4cnc(O)s4)=O)CC3)CCCC2)=O)CC12CC(F)(F)C2 12079,C12(C(CNC(CC3CC(C)C3)=O)NC(=O)CC3CCCOC3)CCC(CC1)C2 12080,N1(C(c2cccc(SCC)c2)=O)CCC(CO)C(NC(=O)Cc2csnc2C)C1 12081,CC(C)(C)C(C(=O)NCC(O)CF)NC(c1ccc(CC#N)cc1)=O 12082,C1(CN)CCCCN1Cc1cccn1CC1CCC(C(=O)OC)O1.n1(C)ccnc1 12083,c1(C2(NC(=O)OCC3CCCCC3)CC2)ccc(OC(F)F)cc1 12084,c1(C(=O)NCCN(C(C)C)C(C2(CCN(C)C)CC2)=O)cc(C(F)F)ccn1 12085,C(=O)(C#CC1CCCCC1)N1CCCCC(NC(c2c(C(C)=O)cn(C)n2)=O)C1 12086,N1(C(CSCC=C)=O)CC2(CNC(C3(C)C=CCC3)=O)CCC1CC2 12087,c1(C(=O)NC2(C)CN(C(=O)Cc3ccsc3)C2)nc2n(c1Br)CCC2 12088,c1(C(N2CCCC(NC(c3ccco3)=O)(CO)C2)=O)c(F)cc(F)c(O)c1F 12089,CC(CC(C)(C)C)C(F)C(=O)N1CCC1CNC(=O)CC1CNC(=O)O1 12090,C1(C(N2CCN(C(=O)CCc3cncn3C)C(C(C)O)C2)=O)CCC2(CCC2)CO1 12091,c1(OC)ccc(S(=O)(=O)N2CC(NC(=O)CCc3cncnc3)C3(CC3)C2)cc1 12092,CC(CC(=O)NC1CCCCC1NC(=O)CC(F)F)S(=O)(=O)c1ccc(F)cc1 12093,C(=O)(C1CCc2nccn21)NCC(C)(C)OCC(=O)Nc1cccc(N(C)C)c1 12094,Cc1cc(C(=O)NC(CNC(c2ccc(CC(N)=O)cc2)=O)C2CC2)ncn1 12095,c1(-c2cn(CC3N(C(C(C4CC4)SC)=O)CC3)nn2)ccc(-c2cn[nH]c2)cc1 12096,c1ccc(F)c(Cl)c1.N1(C(C)=O)CC(C)(n2c(=O)ccc(=O)[nH]2)C1.C1CC1 12097,c1(C(N2CCC(CC=C)(NC(C3CC(C)OC3C)=O)C2)=O)cnc2nccn2c1 12098,Cc1nnccc1C(N1CC2CC1C2NC(=O)COCCc1cccs1)=O 12099,N1(C(C2=CCCN(C(C3CCC(C)O3)=O)C2)=O)CCCC(C2(C)CC2)C1 12100,c1(OC)ccc2onc(CC(=O)NC(C)C(C)NC(c3c[nH]c(=N)o3)=O)c2c1 12101,C1(CNC(CC2(C)CC2)=O)CCCN(C(c2ccc(-n3cnnc3)cc2)=O)CC1 12102,c1(CCNC(=O)CSc2cc(Cl)ccc2Cl)cc(Cl)c(Cl)cc1F 12103,N1(Cc2cc(C)n(CCC)c2C)CCS(=N)(=O)C(C)(C)C1 12104,c1(C(=O)NC(C(C)NC(c2nccc(C)c2)=O)C)cc2c[nH]cnc-2n1 12105,C1(NC(C(C)CN(C(=O)CCCCC#N)C)=O)CCC(=O)N(C)C1=O 12106,C1(=O)C(C(CC)CC)N1.C(C)(C(=O)NC)N(CC(C)C)CC=C 12107,N1(C(c2c(OC)cnnc2OC)=O)CC2ON=C(CNC(c3ccco3)=O)C2C1 12108,N1(C(C2CCN(CC)C2)=O)CC(C(=O)NC2CC(=O)N(O)C2)CC(C)C1 12109,CCC(C(=O)N1CC(O)(CN(C)C)C1)N(C)C(C1CCC1C#N)=O 12110,n1(CC(=O)NCC(C)N(C(CCC(C)SC)=O)C)c(=O)cnc2ccccc12 12111,c1ccc2cc(C3(NCCSC4CCCO4)CCC3)ccc2c1 12112,C1(CC(=O)NC)CN(C(c2ccn(C(C)C)n2)=O)CCN1C(=O)COCC(C)C 12113,c1(C(=O)NC2C(NC(=O)CSCc3ncc[nH]3)CCC2)cccc[n+]1[O-] 12114,N1(C(=O)OC(C)(C)C)CCC(C)(C(N2CCC(OCC3CCCO3)CC2)=O)C1 12115,c1(C(N2CC3C(CNC(=O)C(C4CC(F)(F)C4)O)C3C2)=O)ccc(O)c(Cl)c1 12116,N1(C(CC=C)=O)CC(C(=O)N(CC2=CCSC2)C)C2(CCC2)C1 12117,C1(NC(C(C(C)C)O)=O)C2CC3C1C3C2C(=O)NCc1ccccc1F 12118,c1(C(N2C(C(C)NC(C(C)=CC)=O)CCC2)=O)ccc(CO)cn1 12119,c1(CC(=O)NC(C)(C)CNC(=O)CC2CC3(CC3)C2)c[nH]c2ccccc2c1=O 12120,c1(OC)cccc(C(C(=O)NCCCCC(C)NC(=O)C(C)CN(C)C)OC)c1 12121,N1(C(C)C)CCCC(C(=O)Nc2scnc2C(=O)NC(C2CCOC2)CNC)C1 12122,CC1(C)C2CC=C(CCOC(C3CC3c3cc(Cl)cc(Cl)c3)=O)C1C2 12123,N1(C(C2CC(NC(C=C(C)C3CC3)=O)C2(C)C)=O)CCN2CCCC2C1 12124,n1(CC(N2CCC(NC(CC3C(C)=NOC3=O)=O)C2)=O)cc2ncccc2n1 12125,c1(CN(CCCC)C(=O)NC2CNCCOC2)ccc(C2CC2)cc1Cl 12126,C1(O)(C(C(=O)NCc2ccccc2)NC(C2CS(=O)C2)=O)CCCCC1 12127,C1(CC)C(NC(C2CS(=O)C2)=O)CCCN1C(c1ccc(C)c(C)c1)=O 12128,CC1CCc2c(C(N3CCCCC3CNC(c3cccc(=O)n3C)=O)=O)n[nH]c21 12129,CC(C)C(C(C)NC(c1cscc1Cl)=O)NC(c1ncoc1-c1ccon1)=O 12130,CCCS(=O)(=O)C(C)C(=O)NC1CC(CNC(C2CN(C)CCN(C)C2)=O)C1 12131,c1(C(N2CCC3(NC(=O)CNS(=O)(=O)C4CC4)C(C2)C3)=O)n[nH]c2c1CCCC2 12132,C1(CNC(CCc2cc(C)no2)=O)CCN(C(c2cc(Cl)c(Cl)n2C)=O)CC1C 12133,N1(C(C(c2c(C)n[nH]c2C)C)=O)CC(NC(c2conc2C2CC2)=O)CC(C)C1 12134,c1(C(N2CCOCC2c2cccs2)C(=O)NC2CCCC2)cccc([N+](=O)[O-])c1 12135,CCC(CC1CCCCC1)C(=O)N(CCNC(C)=O)CCNC(=O)C(C)SC 12136,C1(C(=O)NCCC(F)(F)Cn2cc(-c3cncc(C)n3)nn2)(CC)CCCOC1 12137,C1(C(=O)NCC(=C)Br)COC2(C1)CN(C(=O)C(C)OC)C2 12138,c1(C(N2CCC(O)(CNC(CCC(C)OC)=O)C2)=O)ccnc(C)c1C 12139,C1(NC(C2CCC(O)C2)=O)CC2(CCN(C(C3(F)CC=CCC3)=O)CC2)C1 12140,C(=O)(C1=NN(c2ccc(F)cc2)C(=O)CC1)Nc1ccccc1.CC1C(C)(C)N1 12141,n1(CCC)cc(C(=O)N(CCNC(=O)CC2OCCC2C)C(C)C)nn1 12142,c1(C(=O)NC(CC)CNC(=O)C(C)SC(F)(F)F)ccc([N+](=O)[O-])s1 12143,N1(C(C(CC)F)=O)CC23CCCCC2(C1)CN(c1nccnc1C#N)C3 12144,Cc1ncnc(C)c1CC(=O)N(CC(O)CNC(c1occc1CN(C)C)=O)C 12145,c1(C(N(C2CN(C(CCCN(C(C)=O)C)=O)C2)C)=O)ccc([N+](=O)[O-])s1 12146,C1(NC(C2CCC(CC)O2)=O)CC(OC)CN(C(=O)CCc2ccn(C)c2)C1 12147,Cc1nc2cc(C(=O)NC(CNC(=O)CN3CCCCC3=O)CO)c(F)cc2[nH]1 12148,C=CCC(C(=O)N1CC(SCC)C1)NC(c1ccnn1CCC)=O 12149,Cc1cc(C(=O)NC2CC(CNC(C3CC3(C)C(C)C)=O)C2)c(F)cc1Cl 12150,c1(C(C)C)cc(C(=O)NC(C)CN(C)C(c2cc(N)c(F)cn2)=O)cc(O)n1 12151,C1(CN(C(C2C(C(=O)OCC)CC2)=O)C)CC(F)CN1C(c1c[nH]nc1C)=O 12152,C1(CC)CCC(N=c2ccc(Br)c(S(=O)(=O)NC(c3cccs3)C)[nH]2)CC1 12153,N#CC1(C(=O)NCC(CO)NC(C2CN3CCC2C3)=O)CCCCC1 12154,CC1CCC(C(=O)N(C(c2cn(-c3ccccc3C(=O)O)nn2)C(C)C)CCO)OC1 12155,C1(NC(C23N(C(CN(CCOC)C)=O)CCC2C3)=O)CN2CCC1(C)CC2 12156,C(=O)(C(C)(C)C(C)C)NCC(C1(O)CN(C(CSC(C)C)=O)C1)(C)C 12157,N1(C(C(CC=C)CC)=O)CC(NC(C2CC(C)(C)C2)=O)CC2(CCC2)C1 12158,N1(C(CCn2c(C)cc(C)n2)=O)CCC2CC1CN2C(C1CCCS(=O)(=O)C1)=O 12159,Cc1cc(C)c2[nH]c(=NCC(C)NC(=O)Cc3c(F)cccc3Cl)sc2c1 12160,C(CO)(CC(C)CC)NC(CSCCNC(C(C=C)C)=O)=O 12161,c1(CCC(=O)NC(CN(C(=O)C(C)CC(F)F)CC)C)c(C)ncnc1O 12162,N1(C(COCC=C)=O)CC2C=CC1C(C(=O)NCC(CO)C(C)CC)C2 12163,N1(C(=O)CCOc2ccc(F)cc2)CCN(C(=O)Cn2ncnn2)C2CCCC12 12164,c1(C(=O)NCC(C)N(C(=O)CC2SC(=N)NC2=O)C)ccc(O)nn1 12165,CN1CCC(C(=O)NC2(C3CN(C(=O)CCc4n[nH]c(=N)s4)C3)CC2)CC1=O 12166,C1(CC)CCCC1C(=O)N(CC(C)CNC(c1csc(C)c1)=O)C 12167,Cc1ccc(F)c(N)c1C(N1CC(NC(C23CC(C2)C(C(F)(F)F)O3)=O)C(C)C1)=O 12168,Cc1sc(C)c(C(=O)NCC2CCCCC2NC(=O)CSc2cn[nH]c2)c1C#N 12169,c1(CC)nc(-n2cccc2)sc1C(=O)NC1CN(C(c2cnoc2C)=O)CC1C 12170,CN=c1[nH]c(=NC(C)c2cccc(S(N)(=O)=O)c2)[nH]c(=NC(COC)C2CC2)[nH]1 12171,c1(C(=O)NC2(CCNC(C3(COC)CC3)=O)CC2)ccc2c(c1)COC2=O 12172,N1(C(c2ccc(C)s2)=O)C2CCC1CC(CNC(c1ccn3cccc3c1)=O)C2 12173,Cc1occc1C(=O)NCc1cn(C(c2ccccn2)C)nn1 12174,Cc1[nH][nH]c2ncnc(=NCC3(CNC(C4C(C)C4C)=O)CCC3)c1-2 12175,c1(C(C)C)nc(C(=O)NCC(C)(C)NC(c2cc(C(N)=O)no2)=O)cs1 12176,CS(=O)(=O)c1ccccc1CNCC1CC2CC1CC2(F)F 12177,N1(C(C(C)(C)NC(=O)OC(C)(C)C)=O)CC=C(c2cccs2)C1 12178,C(=O)(CC1COc2ccccc21)NC1C(CNC(CC2(C=C)CCOCC2)=O)C1 12179,c1(C(=O)NCCC2(NC(=O)CCNC(N)=O)CC2)cnc(-c2ccco2)s1 12180,c1(CCNC(N2CCCC2C2CCCC2O)=O)cccc2n[nH]cc12 12181,C(C(=O)N1CCC(N2CCC2)C1)(C(C)(C)C)NC(C(C)=C(C)C)=O 12182,C1(CNC(Cn2c(=N)scc2)=O)CN(C(=O)CSC(F)(F)F)CCO1 12183,N1(C(C(CCSC)O)=O)CCC(CNC(=O)C(c2cnccn2)C)CC1C 12184,c1(C(C(=O)NCCSC)N(C)Cc2c(C(=O)OC)cccc2)ccc(F)cc1Cl 12185,CC1CN(c2cc(C(F)F)ncn2)CCC1NC(C1CCC2CC2CC1)=O 12186,C1(C(N2CC(NC(c3cc(C)no3)=O)C(C(F)F)C2)=O)CCn2c(O)nnc2C1 12187,C1(CC(=O)OC)CS(=O)(=O)CCN1C(=O)C(=O)N=S(C)(C)=O 12188,c1(C(=O)OC)ccc(C(=O)NCC(C)NC(=O)CCN2CCNC(=O)C2)c(Cl)c1 12189,C1(C(=O)NC(c2ccccn2)C#N)C2CN(C(=O)Cc3ncccn3)CC12 12190,CC1(NC(c2cnn(CCNC(c3ccccc3C#N)=O)c2)=O)CCC(O)CC1 12191,Cc1noc(C)c1CNC(C1CCN(C(C2CCC(O)C2)=O)CC1)=O 12192,C1(CNC(c2ccccc2Cl)=O)CCCC12CN(C(=O)Cc1ccsc1)C2 12193,C1(C(=O)NCC2(OC)CCN(C(C34CSC(C3)C4)=O)C2)CCS(=O)(=O)CC1 12194,C1(CNC(C2C(C)OC(C)C2C)=O)CCC2(CN(CCOC3CCCCC3)C2)O1 12195,C(c1ccc(C(=O)NC2CC2CNC(=O)C(C)(C)CO)o1)=CC(=O)OC 12196,N1(C(c2ccn(CCOC)n2)=O)CCN(C(c2c(C)ncn2O)=O)CC2(CC2)C1 12197,CCC(C(=O)OC)C(=O)NC1CCCCN(C(C2OC(C)CC2C)=O)C1 12198,N1(C(=O)CC2CCCC2(F)F)CCC2(C1)CN(C(=O)Cn1ncnn1)C2 12199,N1(C(C(c2cn(C)nn2)NC(=O)CC2CSCCO2)=O)CC2CC1C(F)(F)C2 12200,CC1CCCc2nc(C(=O)N(CC(O)CN(C(=O)Cc3csc(S)n3)C)C)cn21 12201,c1(C(=O)NCC2(OC)CCCCCC2)ccc(F)c(-c2nn[nH]n2)c1Br 12202,C12(CNC(C3OCCN(C(C)=O)C3)=O)CCC(CC1)N(C(c1cnoc1C)=O)C2 12203,C1(CNC(C(=O)N(c2ccccc2O)C)=O)CC2CN(C(c3nncn3C)=O)CC12 12204,c1(-n2c(CCCCSC)nc(-c3ccc(F)cc3)n2)ccc(F)c(Cl)c1 12205,C=C(C)C(CC(=O)N1CC(OCCNC(=O)C(c2cnn(C)c2)C)C1)OCC 12206,N1(C(C2CCC(CC)O2)=O)CCC2(CCC(NC(c3cn(C)nn3)=O)CC2)C1 12207,N1(C(C(CCC)C#N)=O)CC2CCC1C1CN(C(=O)COc3cccnc3)CC21 12208,C12(C(N3C(CCC(=O)NC)CCCC3)=O)CCC(C)(CC1)O2 12209,c1(CS(=O)(=O)N(CCNC(C=CC)=O)C2CC2)cccc(OCC)n1 12210,N1(c2cccc(-c3cnc(C)[nH]c3=N)n2)CC(C)CCCC1C 12211,N1(C(c2c(CNC(c3cnc(CC)s3)=O)ocn2)=O)CCCN(C)CC1 12212,c1(C(=O)NC(CCOC)CNC(=O)C=CC2CCCC2)cnc[nH]c1=N 12213,c1(NC(CCC=CCC=C)=O)ccc(NC(=O)C(O)P(C)(C)=O)cc1C 12214,N1(C(c2c(CCC)[nH]cc2)=O)CC2CC(C1)N(C(=O)Cc1cc(O)nnc1O)C2 12215,c1(NCC(CCCC)NC(=O)CC2CSCCS2)nc(Cl)ncc1C(C)=O 12216,N1(C(CSCCC#N)=O)CC23COCC2(C1)C3C(=O)O 12217,c1(OC)ccc2cc(C(=O)NCCCOCCNC(=O)C(C)OC3CC3)[nH]c2c1 12218,c1(CC(=O)N(CC)CC2CCCN2C(=O)CC2OCCCO2)ccc(F)c(C)c1 12219,CS(=O)(=O)c1ccc(CC(=O)NC2CC2(C(=O)O)C(=O)O)cc1 12220,C1(C(=O)NC(CCC)CCC)CCCCN(C(=O)CC2C=CCCC2)C1 12221,c1(C(=O)NCCCOCCNC(c2cc(CC)sc2)=O)nccn2nccc12 12222,c12ccccc1CNC(=O)CS2.C(=O)(C(C)(C)OC)N(CCOC)CC 12223,N1(C(c2c(CC)noc2)=O)CCC2(NC(c3occ(C)c3C)=O)CCCCCC12 12224,C1(C(=O)NC2C(C(=O)NCC3(OCC)CN(C)C3)CCOC2)C2CCC(C2)C1C 12225,C12(C(=O)Nc3cc(C)nn3C)CCC(C(=O)NC(c3cnccn3)C)(CC1)C2 12226,C1(NC(=O)CCF)(CNC(C2CCC(N3CCOCC3)CC2)=O)CCCCC1 12227,C1(N(C(=O)C(C2CC2)N(C)C)CCOC)CCN(C(C2CS(=O)(=O)C2)=O)CC1 12228,C1(NC(CCN(C)CCO)=O)CCN(C2CCN(C(C3CC=CCO3)=O)C2)CC1 12229,Cc1cccc(Br)c1C(=O)Nc1ccsc1C(=O)Nc1c[nH]nc1C#N 12230,c1(NC(C2CN(c3ncnc4ccsc34)CCC2O)=O)ncc2c(n1)CCC2 12231,CC(C(=O)N(C1CC(C(=O)N(C)CCN(C)C)C1)C)OCC1(CO)CC1 12232,C(=O)(C(F)CCC)NC(c1ccccc1)CNC(CCOCC#C)=O 12233,N1(C(C(CC)OC)=O)CCC(CC(N2CC(C(C)C)C2)=O)C1(C)C 12234,CC(C)(C)C#CC(=O)NCC1CCCCC1C(=O)NOCCC(F)F 12235,c1(OC)ccc(NC(=O)NC2CCCCCC2)c(C(=O)N(C(C)CO)C)c1 12236,c1(C(=O)NC2CCCN(C(CCCCOC)=O)C2)cnc2c(cnn2C)c1 12237,CC1CCN(C(=O)C(c2ccc(F)c(F)c2)(C)C)CCN1C(C1CCCOC1)=O 12238,C(C(C(F)F)c1nc[nH]n1)NC(=O)CNC(c1ccccc1)c1ccccc1 12239,N1(C(CCC(C)C)=O)CC(O)(C2(CNC(c3cccc4ccnn34)=O)CC2)C1 12240,Cc1c(C(=O)N(CC(C)(C)NC(=O)C=CCO)C)[nH]c2c1CCCC2 12241,C(=O)(CC1=NNC(=O)C1)N1CCN(C(c2c(C)oc(CCO)c2)=O)CC1CO 12242,N1(C(C2(CCC)CC2)=O)CC(NC(=O)C(=Cc2ccc(C)cc2)C)C2(CCC2)C1 12243,CC(CF)CC(=O)NCCCC1(NC(c2nccnc2N)=O)CC1 12244,Cc1nscc1C(=O)NC(C1CCN(C(=O)CC2CCCN2C(C)C)C1)(C)C 12245,CC1CC2CN(C(C3CCC(NC(=O)CC4CCCO4)C3)=O)CCN2C1 12246,Cc1nc(=NCC2CCC(NC(c3ccc(N(C)C)cn3)=O)C2)[nH]cc1[N+](=O)[O-] 12247,c1(OCC)nc(NC(C(C)NC(c2cc(COC)cs2)=O)C(C)C)ncc1Cl 12248,C1(C(=O)NC2(CO)CN(C(c3ccc(C)c(Br)c3)=O)C2)CCn2ccnc2C1 12249,Cc1cn2cc(NC(c3cscc3-c3cccc(CO)c3)=O)ccc2n1 12250,CC(CC(=O)NCC1(C(C)(C)O)CN(C(=O)C(C2CCCCC2)O)C1)P(C)(C)=O 12251,[N-]=[N+]=NC1CCN(C(=O)C(C2CCCO2)NC(=O)CSC2CC2)CC1 12252,c1(OCCOC)ccc(CN(c2ccc(C(=O)O)c(C)c2)C)cc1OC 12253,C(=O)(CCN(OC)C(=O)CS(=O)C(F)(F)F)N1C(CC)CC1C 12254,N1(C(c2ccc(C)c(C)n2)=O)CCC2(CCCN(C(c3cnc(=N)[nH]c3)=O)C2)C1 12255,C12(NC(C(c3cccc(Cl)c3)CC)=O)COC(C)(C1)C2 12256,c1(CC(=O)NCC(CC)(CC)NC(C2CNC(=O)N2)=O)c[nH]c2ccc(C)cc12 12257,C1(C(=O)NCc2cc(C)on2)CCC(NC(=O)Cc2ccccc2Br)CC1 12258,C1(CC=C)(NC(=O)CNC(=O)OC)CCCN(C(=O)C=Cc2cccc(Cl)c2)C1 12259,C1(NC(C(C)C)=O)CCCCCC1C(=O)NCCCOC(=N)O 12260,C=C(Br)CC(C)(C)C(=O)NC1CCCN(C(C2(C#N)CCOC2)=O)CC1 12261,C1(NC(c2nc(CCC)oc2)=O)CCC(C(=O)NC2C(C)CCC2C)CC1 12262,C1(CC(=O)NC2C3CN(C(C4CCN(C(C)=O)CC4)=O)CC32)CCC2(CC1)CC2 12263,N1(C(=O)CC2CCCC3CC23)CC(C2CC2)(C(N2CCCC(CCO)CC2)=O)C1 12264,c1(CC)cnc(C)c(NC(=O)C(CCNC(=O)CP(C)(C)=O)OC)c1 12265,c1(OC)nsc(OC)c1C(=O)NCCC(C)N(C)C(c1ccc(OC)cc1)=O 12266,c1(C(N2CC3(CCCCN3C(c3ccns3)=O)C2)=O)cc2cc(F)cc(F)c2[nH]1 12267,C(=O)(N=c1cc2ccccn2[nH]1)C1N(C(Cc2c(C)n[nH]c2)=O)CCSC1 12268,C(CCN=C(NCCC1=CCOCC1)N1CC(C)S(=O)(=O)C(C)C1)OCCOC 12269,CCC(C)(C)C(=O)N(C)CC1CCN(C(c2cnc(SC)nc2)=O)C1 12270,C#Cc1cccc(C(N2CC(CC=C)(NC(C3CCCC3(C)C)=O)C2)=O)c1F 12271,N1(C(CC#N)=O)CCC2CCN(C(=O)CCn3ccnc3)CC2C1 12272,C1(C(N2C(C)C(NC(c3cc(O)nn3C)=O)CCC2)=O)CCc2cnn(C)c2C1 12273,N1(C(CC(C)NC(=O)CCc2ccn(C)c2)=O)CCOCC1CCO 12274,C(CC(F)F)(C(=O)NC(c1cccs1)C)NC(Cc1cc(C)nn1C)=O 12275,c1(SC)ncc(N)c(C(=O)NCC2CC(F)CN2C(=O)CN(C)C2CC2)n1 12276,N1(C(C(c2ccccc2)NC(C)=O)=O)CCC(C)(NC(=O)CC2(O)CCC2)C1 12277,Cc1oc(Cl)nc1C(=O)N(C(C)CCNC(=O)Cc1ccccc1O)C 12278,C12(C(N3C(C#C)CCC3)=O)C(NC(C3CCC(N(C)C)C3)=O)C3CC1C2C3 12279,C1(C)(CC)CCC(C(=O)N(C2(CC(=O)NC(C)(C)CCCO)CC2)C)O1 12280,C1(C(NOC(C=C)C)=O)CSCCN1C(c1ccsc1Cl)=O 12281,CN1CC(C(N2CCCC(NC(=O)CCCc3ccsc3)C2)=O)CC1=O 12282,C(=O)(C1=C(C)CCCC1(C)C)N1CC(CNC(C(CCCC)(C)F)=O)OCCC1 12283,c1(CC(C)NCc2ccc(Cl)cc2)ccc(C#N)cc1 12284,C1(NC(c2c(CC)nn(C)c2)=O)C2CC3CN(C(=O)CC4CN(C)C4)C1C3C2 12285,c1(C(N(CCOC)CCNC(c2cccnn2)=O)=O)c(O)ncc(Br)c1C 12286,N1(C(C(=O)NCC2COC(C)(C)O2)=O)CCOC(C(F)F)CC1 12287,C(C(=O)N(CCC(=O)N1CCC(F)(F)C(C(N)=O)C1)OC)(C1CC1)OC 12288,Cc1cc(C(=O)NC(C(N2CCCC2CF)=O)C2CC2)sc1C 12289,C1(NC(c2cc(CCC)on2)=O)CCCN(C(c2cnn(C(C)C)c2)=O)CC1 12290,C1(NC(C(c2ccccc2F)(C)C)=O)CCN(c2nnc(CO)o2)CC(O)C1 12291,N1(C(c2ccn(C(C)C)n2)=O)CCCC(NC(=O)CC2COCCN2C)C1 12292,Cc1ccc(OCC(=O)NCC2CCCN2C(=O)Cn2ncccc2=O)c(C)c1 12293,c1(CC)cc(C(=O)N(CCCN(C(=O)CSC(F)F)C)C)sc1C 12294,C1(NC(C(=O)NCCCOC(C)=O)=O)CCOCC1 12295,C1(CNC(COC)=O)CC2CCC1N2C(c1cc(C)cc(C)n1)=O 12296,N1(C(CC2CC(CC)C2)=O)CCOC(C)(CC)C1.C12(CCN(C)C1)C(=O)N2 12297,Cn1c(C(c2ncccc2O)(C)O)nnc1C1CCCN(CCCOC(=N)O)C1 12298,N1(C(C(=O)NCC(F)(F)C2CCC2)=O)CCC(O)C(F)C1 12299,CCCCC(C(=O)NCCn1cncn1)NC(c1cn[nH]c1)=O 12300,S(=O)(=O)(c1cnc(N(C)Cc2ccnn2C)cc1C)NC1CC(CC)OCC1 12301,CCCC(CC)CCC(=O)NC(CNC(=O)CCN(C)CC)C1CCC1 12302,c1(CNC(N2CCC(C(N(C)C)=O)C2)=O)ccc(N2CCCS2(=O)=O)cc1 12303,Cc1cc(C(=O)NC(CNC(C2(CC3CC3)CC2)=O)C2CC2)n[nH]1 12304,N1(C(C2CCN(C3CC3)C2=O)=O)CC2(CCN2C(c2ccc([N+](=O)[O-])[nH]2)=O)C1 12305,CC1(CNC(c2cnccn2)=O)CCN(C(c2c(Br)cnn2C2CCC2)=O)C1 12306,S(=O)(=O)(c1ccc2c(c1)CCCC2)CC(c1ccnc(OC(F)(F)F)c1)=O 12307,C1(CNC(C=CCC)=O)CCC2(CN(C(=O)C(c3ccccc3)SC)C2)O1 12308,C1(NC(CC(CC)C)=O)CC12CCC(NC(c1cccnc1C(F)F)=O)CC2 12309,c1(C(=O)NC2CC(NC(C(CCC)O)=O)C(O)C2)cccc2ccc(C)nc12 12310,c1(C(N2CC(O)(C3CC3)C2)=O)cc2c(F)c(Cl)ccc2[nH]1 12311,c1(OC(=O)NOC2CN(Cc3cc(Br)co3)C2)ccccc1 12312,N1(C(c2cnc(CC)s2)=O)CCCC(CNC(c2ccc(C#N)s2)=O)C1 12313,N1(C(C=CCC(C)(C)NC(CC(C=C)CC)=O)=O)CCN2C(=O)NCC2C1 12314,c1(CC)nc(C)n(C)c1C(=O)NCCCOCCNC(C1CCC2(CC1)CC2)=O 12315,C1(CCC)CN(C(c2cnns2)=O)CCN1C(=O)CN(C)C(c1cccs1)=O 12316,Cc1ccc2nc(SCC(N3CC4CCN(C(=O)C(C)CO)CC4C3)=O)[nH]c2c1 12317,c1(SC)nc(NC23CCC(CC2NC(=O)CCCCCSC)C3)cc(C(F)F)n1 12318,C(CCC(=O)N(C)CCN(C)C(c1cc(-c2cccs2)[nH]n1)=O)OCC 12319,N1(C(C(C)SC(C)C)=O)CCC(C)(C)C1CC(=O)NCC1CCCCC1 12320,C1(CCNC(CC2(OC)CC2)=O)(NC(=O)CCCc2cccs2)CCCC1 12321,N1(CCC(=O)NCC2(CN(C(C(CC)C)=O)C)CC2)CCCCC1C 12322,N#Cc1ccccc1C1CN(C(c2c(C(=O)O)cccc2C(=O)O)=O)C1 12323,C1(C)(CCN(C(=O)NCCOCCOCCC#C)C2CC2)CC(F)(F)C1(F)F 12324,N1(C(C2CC(OC(C)(C)C)C2)=O)CCC(O)(CCNC(C2CCSC2)=O)CC1 12325,C(c1cncn1C)=CC(=O)NCC1(CN(C(C(C)OCC(F)(F)F)=O)C)CC1 12326,c1(CN2CCC(C(=O)NCc3ccc(OC)cn3)C2)ccc(F)c(F)c1 12327,CC1CCOCC1COC(C1(Cc2ccccc2Cl)CCCCC1)=O 12328,c1(CN(CCNC(C(c2ccc(N)cc2)OC)=O)CCOC)ccccc1Cl 12329,c1(CN2CCC(NCc3ccc(C(F)(F)F)cc3)C2)cc(N)c(Cl)cn1 12330,CCC(C(=O)NCCOCCNC(c1ccc(N)c(Br)n1)=O)C(C)(F)F 12331,C(=O)(CC(C)C(C)C)N1CCC(C(=O)NC(C(=O)OC)(C)CO)C1 12332,c1(C(=O)NC2CCN(C(=O)C3=COCCC3)CC2O)cnc2ccc(F)cc2c1 12333,c1(C(N(C2CCN(C(c3c(CC)nc[nH]3)=O)C2)C)=O)nc2cnccc2s1 12334,CCC(C)(C)C(O)C(=O)NC1(CCNC(=O)CC2CCC(C)(C)C2)CCC1 12335,CCC(C)C(O)C(=O)N1CCCC(C)(CNC(=O)CC2CC(F)C2)C1 12336,c1(C(=O)NCC(C(C)C)NC(C2(C)CSC2)=O)cc2cc(F)cc(F)c2[nH]1 12337,C1(NC(COCc2onc(C)n2)=O)CN(C(=O)C(C)Cc2ccncc2)CC1F 12338,CCC(CC(=O)N(C1CC(NC(c2cc(Cl)ns2)=O)C1)C)C(C)(C)C 12339,C(=O)(C(CC)(CC)CO)NCC1N(C(CNC(C(CC)C)=O)=O)CC(F)C1 12340,c1(C(=O)NC(CNC(c2cc(C)nnc2)=O)C2CCC2)cc([N+](=O)[O-])ccc1N 12341,CCC(CC(F)F)C(=O)N1CC(NC(N)=O)CC(NC(=O)CCOC)C1 12342,N1(C(CN(CCCCCC)C)=O)CC(CNC(C2(CO)CC2(F)F)=O)C(O)C1 12343,N1(C(CCc2c(C)ncs2)=O)CCN2C(=O)C(NC(C34CSC(C3)C4)=O)CC2C1 12344,c1(C(=O)NC2CN(C(c3c(C)cc(O)cc3)=O)C(C)(C)C2)cccc2c1COC2 12345,c1(C(N2CC(O)(C(C)NC(C(CCC)CC)=O)C2)=O)cc(C)c(Br)c(C)c1 12346,C(=O)(C(F)C(F)(F)F)NC1(CC(=O)NC2CCC(C(N)=O)CC2)CCOCC1 12347,C1(N(C(CC2CC(CC)C2)=O)C)CC2CC1N(C(c1csnc1C)=O)C2 12348,c1(C(N2CC(C(=O)NC(C=C)CO)C(F)(F)C2)=O)ccc2nccn2c1 12349,C1(C2CCN(C(C3CCCCCS3(=O)=O)=O)CC2)(NC(C2CCCC2)=O)CCC1 12350,N#CC1(c2ccc(C(=O)N(C3CCNCC34CC4)CC(O)CO)cc2)CCCC1 12351,N1(C(c2cccn(C)c2=O)=O)CC2CCCC(NC(C3CCCSC3)=O)C2C1 12352,c1(C(N(CC(CC)NC(=O)C(C2CC2)OC)C)=O)cc([N+](=O)[O-])n[nH]1 12353,N1(C(C(C)CC2CC2)=O)Cc2ccccc2CC1CNC(=O)C(C)C(C)(F)F 12354,N1(C(C2C(C#C)C2)=O)CC2(CCC2)CC1CNC(c1cnn(C(C)C)n1)=O 12355,C1(C(=O)NC2CCCN(C(C=C(C)CN3CCOCC3)=O)C2)CC2CCC(C1)S2 12356,C1(CN(C(C2(SC)CN(C(=O)CSC(F)(F)F)C2)=O)C)CCCCC1O 12357,C1(CNC(c2c(C)cc(SC)o2)=O)CC2CCCC2N1C(=O)C(C)CC(F)(F)F 12358,C1(OC)CCC(C(=O)N(C(C)(C(=O)NC(C)CC(C)C)C2CC2)C)CC1 12359,N1(C(C(C)C(F)F)=O)CCC(C)C(N(C)C(c2cc(C(F)(F)F)ccc2F)=O)C1 12360,O=C(CC(F)(F)C(F)(F)F)NC1CCCCC1NC(C12CCCC1C2)=O 12361,C#Cc1ccc(CC(N2CCN(C(C)=O)C(CS(C)(=O)=O)C2)=O)c(F)c1 12362,C=CC12CCN(CC1)C2.C1(C(=O)OC)OCCC1NC(=O)C(C)CC 12363,N1(C(CCC#CC)=O)CC(NC(=O)C(O)Cc2ccc(F)cc2)CC12CCCC2 12364,N1(C(CSCCCC)=O)CCC2(CC1)OCCC2NC(=O)CSc1n[nH]c(O)n1 12365,C1(C(=O)NCC(C(=O)NC(C2CCOC2)(C)C)CC2CC2)CC2(CC(=O)C2)C1 12366,c1(C(N(C2CCN(C(c3ccc(C4CC4)nc3)=O)CC2)C)=O)cc(N)nc(Cl)c1 12367,N1(C(CCC=C=C)=O)CCCC(O)(CCNC(=O)CCN2CCC(F)C2)C1 12368,C1(NC(c2ccn(CCC)n2)=O)CCC12CN(C(=O)CCOCC)C2 12369,CCCC(C(=O)NC(C)CC(N)=O)NC(=O)C(C)N1CC(C)C1 12370,C(=O)(C1=CCCC1C)NC(C(=O)NC1CCCN(C(C)=O)C1)CCN(C)C 12371,C12(NC(c3cc(C)c(Cl)cn3)=O)CCCC1CN(C(C1CN(C(C)C)C1)=O)C2 12372,CCC(CC)C(C(=O)N(CCNC(C1(O)CCCC1)=O)C1CC1)N1CCOCC1 12373,N1(C(C(C)=C2CCC2)=O)CCN(CC(=O)N(CC(F)Cl)C)CC1 12374,N1(C(CNC(C2(CC(C)C)COC2)=O)=O)CC(C)(NC(C(N)=O)C2CC2)C1 12375,N1(C(CNC(C2C(CCC)C2)=O)C)CCN(C(=O)Cc2ccn(C)n2)CC1 12376,N1(C(c2cc(C)no2)C(=O)NCC(F)F)CCc2cc(C#N)ccc2C1 12377,c12ccc(cc1)NC2C.Cc1nccn1Cc1nccn1C 12378,Cc1nc(Br)ccc1CNC(c1ccc(NS(=O)(=O)C(F)(F)F)nc1)C 12379,N1(C(CC=CC)=O)CCC(C2CCN(C(c3n[nH]c(C4CC4)n3)=O)C2)C1 12380,c1(OC)cc(C(N2CCC(NC(=O)C(Cl)=CCl)CC2C)=O)ccc1[N+](=O)[O-] 12381,C=C(C)CN=C(NCC(C1CCCCCC1)(C)O)NCC1CCC(C2CC2)O1 12382,n1(CC)ncc2cc(C(N3CCCCCC3c3ccco3)=O)c(C)nc12 12383,C(=O)(C(CC(C)(C)C)OC)N1CCCC(CC)C1C(=O)NCc1sc(C)nc1C 12384,N1(Cc2ccc(CNCCc3n(C)ncc3)cc2)CCCCCCC1 12385,C1(NC(C2C(=C)C2)=O)CCCCCCC1NC(=O)CCc1cnc[nH]1 12386,c1(C(N(CC(CC)C)C)=O)coc2c1CN(C(C1CC1C(F)(F)F)=O)C2 12387,C(=O)(C(O)C(C(C)C)OC)NC(CNC(C(CC)N(C)C)=O)COC 12388,C(N=c1[nH]c(N2CCCC(C(N)=O)(N(C)C)C2)nc(=N)[nH]1)C1(OC)CCCCC1 12389,C1(F)(C(N2C(C)(c3ccc(C(F)(F)F)cc3)CCC2)=O)CC2CCC1C2 12390,C1(NC(c2nc(C)sc2Br)=O)CN(C(C2CN(C)CCO2)=O)CC1(C)C 12391,c1(N2CC3C(C(N4CCC(CSC)C4)=O)C3C2)nc(C)cc(C)c1CO 12392,Cc1ccsc1CCCC(=O)NCC(CO)NC(=O)CN1CCCC1 12393,C12(CNC(CS(=O)(=O)NC)=O)CCCC1CN(C(c1cc(C)co1)=O)C2 12394,Cc1csc(=O)n1CC(=O)NC1C2CC1N(C(c1sccc1SC(F)F)=O)C2 12395,c1(C(N(c2ccc(C)c(C)c2)CCC)=O)ccc2cnccc2c1O 12396,C1CCC(=O)NC12CCC2.C1(=CC(=O)NCCC(C)N2CCCC2)CCOCC1 12397,Cc1cnn(C)c1C(=O)NC(C)C(C1CCCCC1)NC(c1ccsc1)=O 12398,C1(CNC(=O)NCc2cc(C(=O)OC)nn2C)CC12CCc1ccccc12 12399,N1(C(c2ccc(OC)s2)=O)CC(NC(C2CC(N(C)C)C2)=O)CC12CCCC2 12400,N1(C(C2(C)CCN(C(Cc3cccc(SC)c3)=O)C2)=O)CCCC(C)(O)CC1 12401,c1(CCC(=O)NCC2CN(C(COC)=O)C(C)(C)C2)c[nH]c2ccccc12 12402,C(=O)(C1=NNC(=O)C1)NCCCC(C)NC(C1C(CC(C)C)C1)=O 12403,O=C(C1=CC2(CCN(C(=O)CSC3CC3)C2)C1)NCCc1ccc2c(c1)CCO2 12404,CC1CC(NC(c2cn(CCCC#N)nn2)=O)CN1C(=O)CCC(F)F 12405,N#CCCCCCC(=O)NC1CC2CCC1CC2NC(C1CCS(=O)(=O)CC1)=O 12406,C=CC1CCCC(NC(C2CC(C)(NC(=O)C=CC(C)CC)C2)=O)C1 12407,N1(CC)CCN(C(c2nc(Cl)cs2)C(=O)Nc2ccc(Cl)cc2F)CC1(C)C 12408,C(=O)(CCCC(=O)N1CCC(C(C)NC(=O)CC2CCC(C)(C)CC2)C1)OCC 12409,c1(C2CCN(C(CSCCOC)=O)CC2)ccccc1NC(=O)C(C)C1CC1 12410,N1(C(COC(C2CN(C)CCC2O)C)=O)C2CCC(C2)C1C(=O)OC(C(C)(C)C)=O 12411,C1(CNC(=NCC)NCCC(C)(C)C)CC2(CC2)S(=O)(=O)N1 12412,Cc1ccc(C=CC(N2CCC3(CC3NC(=O)CSC(F)F)C2)=O)cc1 12413,C(=O)(C1=NOC(C(C)(C)C)C1)NC(C1CN(C(=O)Cc2cnccn2)CCO1)C 12414,C1(NC(COCCC#C)=O)CCCOC12CCN(C(C1(O)CC1(C)C)=O)CC2 12415,Cc1cccc2c1OC(c1nc(N3CC(C)C(O)C(C)C3)no1)C2 12416,N1(C(C2(CNC(C3CC(=C)C3)=O)CCCO2)=O)CCN(C)C(CC)C1 12417,c1(C(N(C2CCN(C(=O)COc3ccccc3)C2)C)=O)c(N)cnn1C 12418,c1(CNC(CC=C=C)=O)nc2c(s1)CCN(C(C1CC1F)=O)C2 12419,C(=O)(CCCCC(C)C)NC1C2(CN(C(c3cnc(CC)s3)=O)C2)CC1 12420,C(N=c1nc2c(ncn2C)c(N(C)Cc2ccoc2C)[nH]1)C1(CCC)CC1 12421,c1(C(=O)NC(c2c[nH]c3ccccc23)C(=O)OC)cc(S(=O)(=O)O)ccc1O 12422,Cn1cc(C(=O)NC2CC2NC(C2(C3CCCO3)CCC2)=O)c2cccnc12 12423,c1(OC)cc(C)ccc1OCC(=O)N(CCC(C)NC(=O)C(C)S(N)(=O)=O)C 12424,S(=O)(=O)(c1c[nH]c(C(N2CCN(C(C3(F)CCCC3)=O)C(C)C2C)=O)c1)NCC 12425,N1(c2nnc(C)s2)CC2(C1)SCCC2NC(C1CC(=O)N(C(C)C2CC2)C1)=O 12426,CC1NC(=O)CCC1NC(=O)C1=NOC(CNC(C2COCCN2C)=O)C1 12427,C1(N2CCC(N(C(=O)CC3CCCCCC3)CC3CC3)CC2)CCC(=O)NC1=O 12428,C12(NC(CN(S(CC)(=O)=O)C)=O)CCN(C(c3ncn4c3CCC4)=O)CC1C2 12429,c1(C(N(C)C(=O)OCCOC(c2ccccc2F)=O)=O)cc(F)cc(Cl)c1 12430,C=CCN=C(NCC(c1cccc(Br)c1)C1CC1)N1CCC(OC(=O)NC)CC1 12431,N#CC1(C(=O)NC2CC(CCNC(=O)C=C(Cl)Cl)C2)CC2(CC2)C1 12432,Cc1c(C(N2CC(NC(C3(C4CC4)CCC3)=O)C2)=O)[nH]c2ccc(C(C)C)cc12 12433,Cc1cnc(C=CC(=O)NCCCC(C)NC(c2sc(C)cc2OC(F)F)=O)[nH]1 12434,N1(C(c2ccnc(F)c2)=O)CCC(F)(F)C(CNC(C23CCCC2C3(F)F)=O)C1 12435,Cn1nc(C(N2CC(O)CC2(C)C(=O)NOCC(O)C(C)(C)C)=O)ccc1=O 12436,C1(CNC(C2(C)CC=CCC2)=O)CC12CCN(C(C13CC(C(F)F)(C1)C3)=O)CC2 12437,c1(N2CCN(C3CC(OC)C3)CC2)cccc2n[nH]cc12 12438,c1(OC)cccc(N2CC3CCC2C(NC(C2CC(=O)N2)=O)C3)c1[N+](=O)[O-] 12439,CP(C)(=O)c1cc(C(=O)NCC2CCCN(C(=O)CNC=O)CC2)ccn1 12440,c1(C(N2C(CNC(c3cnc(C)s3)=O)CC(O)C2)=O)cccc(CO)c1C 12441,C1(NC(COCCSC)=O)CCCC1CNC(=O)CCC1CCN(C)C1 12442,Cn1cc(C(N2CC3CC3(C(=O)NCC(=C3CCCCC3)F)C2)=O)n(C)c1=O 12443,CCC(C)C(C)(O)CNC(C1CCC(C2CC2)N1C(c1cccc(O)c1F)=O)=O 12444,c1(C(C(=O)NCC(c2ccccc2)N(C)C(c2cnco2)=O)O)ccccc1Cl 12445,N1(C(CCCOc2ccc(C)cc2)=O)CC2(CCC2c2nn[nH]n2)C1 12446,CC(=O)CCCC(=O)N(C)CC1CCN(C(=O)COCc2ccnc(O)c2)C1 12447,N1(C(=O)COC2CCCCC2)CCC(CNC(C2(F)CC2)=O)C12CCC2 12448,C12(C(=O)NCC(CNC(C3(CC(F)F)CCC3)=O)OC)CC(C(C)C)(C1)C2 12449,C1(O)(CC(=O)OCC)CCN(C(=O)C(C)c2ccsn2)C1 12450,c12cccc(c1)NC(=O)NC2.N1(CC(C)C)CCC(NC2CC2)C1 12451,C1(CC(=O)NC(Cn2cncn2)C(=O)NCC2CC2Cl)CNC(=O)O1 12452,CC#CCC(CO)NC(C1(N(C(C2CC(=O)C2(C)C)=O)C2CC2)CCC1)=O 12453,C(=O)(C(F)C(=O)NC1CN(C(=O)Cc2nncn2C(C)C)CC1C)OCC 12454,C(=O)(N=c1[nH]onc1C1CC1)C1CCC(CC(=O)Nc2ccc(Br)nc2F)CC1 12455,N1(C(C)=O)CCN(C(=O)C(Cc2ccco2)NC(=O)Cc2coc(C)n2)C(C)C1 12456,C1(CC=C)(NC(c2cc(COC)on2)=O)CCN(C(C2CSCCS2)=O)C1 12457,C1(CC)C(NC(C2CSC2)=O)CCCN1C(=O)C=Cc1cncc(OC)c1 12458,c1(NC(C=CCCC)=O)ccc(-c2nccnc2OC(=O)C2CC2)cc1 12459,C1(NC(CSc2n(C)ccn2)=O)CCC2(CC1)CCN(C(=O)CC1CC1(C)C)C2 12460,N1(C(C(CN=[N+]=[N-])NC(C2CCCCC2O)=O)=O)CCn2nncc2C1 12461,CC1OC2(C(=O)NC3C=CCN(C(c4c(F)cccc4F)=O)C3)CCC1CC2 12462,c1(C(N2CC(C)C(CNC(c3cc(Cl)no3)=O)CC2)=O)ccc2ncccn12 12463,C1(C(N(CCCN(C(C(c2cccnc2)OC)=O)C)C)=O)CC1C1CC1 12464,c1(NCC(C)OC(F)F)ncccc1S(=O)(=O)NC1CCc2ncsc2C1 12465,c1(CC)c(C(N2CCN(C(c3cnc(S)[nH]3)=O)C(CCOC)C2)=O)cccc1C 12466,N1(CCCNC(C(CC2CC2)OC)=O)CCN(C(C2(CC3CC3)CC2)=O)CC1 12467,C=CC1(CC(=O)NC2(CC(C)(C)C)CC2)CN(C(C2CC(C)(C)CO2)=O)C1 12468,C1(C(=O)NCC(c2ccccn2)C)CC2CC2N1C(=O)C(C)SN1CCOC1=O 12469,C(CCc1ccc(F)cc1)(C(=O)NCCCC1CC1)N(CCOCCC)C 12470,C=CC1(C(=O)NC(c2nn[nH]n2)C2CC2)CCN(C(=O)C=CCC)C1 12471,c1(C(N(CCCNC(CC(N2CCCCC2=O)C)=O)C)=O)ncccc1Br 12472,CC1CCC(C)(C(=O)N(CC(C)CNC(=O)C(O)Cc2ccccc2)C)C1 12473,c1(C(=O)NCC2CC(NC(c3cc(SC)c(C)o3)=O)C2(C)C)ccc(N)cc1Cl 12474,CC1C(C(=O)N(C2CCOC2=O)C)CCCN1C(c1ccc(F)cc1)=O 12475,c1(N2CCC(CC=C)C2)cc(Br)ccc1S(=O)(=O)N1CCOCCC1 12476,C1(NC(C(CCC)O)=O)CC2CCC(C1C)N2C(=O)C(C)S(=O)CC 12477,c1(C(N2CC3C(CCNC(=O)CSC(F)(F)F)(CC3)C2)=O)cnc2cc[nH]c2c1 12478,N1(C(c2c(CC)nccc2)=O)CCCC(C)(C(=O)Nc2cc(Br)nc(Br)c2)C1 12479,CON(C)C(=O)CN(C)N1CCOC(COC(F)F)C1 12480,c1(OC)cccc(C(C)NC(=O)NC(C(O)CO)C2CC2)n1 12481,CC1CSCCN(C(c2cnn(CCNC(=O)CC3CC(F)C3)c2)=O)C1 12482,CC1CC(CNC(C2(F)CCCCC2)=O)CN1C(=O)CCc1cscn1 12483,C(CC(O)C(=O)N1CCCC(NC(c2ccnc(C(N)=O)c2)=O)C1)N(C)C 12484,c1(OC)ccnc(NC(c2cnc(-c3cc(O)cc(F)c3)cn2)=O)c1I 12485,C1(C(N2C(C(C)NC(c3ccc(Cl)cn3)=O)CCC2)=O)OCC2COCCC12 12486,C1(C(N2CC(c3cn(CC(=C)CC)nn3)(C(=O)OC)C2)=O)CC2C=CC1C2 12487,C1(NC(C=C(CCC)C)=O)CC2CCC(C1)N2C(=O)C(C(CC)CC)OC 12488,CC(C)C(CN(C)C)C(=O)NC1CCN(C(=O)CCC2CC2)CC1O 12489,C(CNC(C1(Cl)CC1C(C)=O)=O)(CC(=O)NC(C1CN(C)CCO1)C)OC 12490,C(CC(C)(C)C(=O)NCC1(C)CCN(C(=O)COc2ccc(Cl)cc2C)C1)OC 12491,N1(C(C(C(C)C)SC)=O)CCC(C)C(NC(c2cc(C(C)(C)C)n[nH]2)=O)C1 12492,N1(C(C(N2C(COCC)C=CC2)=O)=O)CCC2(CC1)CN(C)c1ccccc12 12493,C1(NC(c2ccc(CC)cc2O)=O)CC(NC(c2ccoc2)=O)C12CCOCC2 12494,CC1COC2(CCC2)CN1C(C1CC2CC1CC2NC(c1cccn1C)=O)=O 12495,C1(CC(=O)NC(C(=O)OCC=C)(C)C)C2CCCC2N1C(=O)CCc1cnoc1 12496,N1(C(=O)CO)CCC2(CC1)CN(C(C1C3CCC13)=O)CCO2 12497,C(CC(C)C)(C(=O)N1CCCC(C)(C(N2CC(O)C(O)C2)=O)C1)NC(=O)OC 12498,C(C(C)(C)CNC(C1(OC(C)C)CCC1)=O)N(C(=O)CCc1conc1C)CC 12499,c1(-c2cc(OC)ncc2)nc(C(N2CCC(C(C)(C)O)CC2)=O)ccc1F 12500,Cc1nc(NC(=O)Cc2ccc(C(F)(F)F)cc2)cnc1Cl.C12CC1CNC2=O 12501,O=C1CN(CC(N2CCC3CC23C(=O)Nc2cnccc2CO)=O)CCN1 12502,CC(C)C(O)C(C)C(=O)N1CC=CC1(C)C(=O)NC1(CC2CCC2)CC1 12503,Cn1nc(C(=O)NCC2CC(NC(=O)C(c3ccc(Cl)cc3)(C)C)C2)ccc1=O 12504,c1(CC)n[nH]cc1C(=O)NCCC1CCN(C(=O)C(O)C2CCC2)C1 12505,Cc1cccc(N)c1C(=O)NC1CCC(NC(=O)CCC2CNC(=O)N2)CC1 12506,c1(C(=O)NCC2CN(C(=O)C(CCSC)NC)C2)cc(C)ccc1OC.CO 12507,C=CCC(C(=O)NC1COCC1CNC(=O)C(C(C)(C)C)NC(N)=O)C(C)C 12508,CC1CC(NC(c2csnc2Cl)=O)CCN1C(C1CN2CCC1CC2)=O 12509,C1(C)(CNC(C(C=CC)O)=O)CC(F)(F)CN1C(=O)CNC(c1ccncc1)=O 12510,c1(C(=O)NCC2C(C)(C)C(NC(=O)Cn3nccn3)C2)ccnc2ccnn12 12511,c1(CCNC(C2CCC(=O)N2CCN2CCOCC2)=O)cccc2cc[nH]c12 12512,c1(C(=O)NCCCC2N(C(c3c(C)ccs3)=O)CCC2)ccccc1OC1CC1 12513,CC1=C(CNC(=O)C(C(C)O)NC(=O)CC2CCCCO2)COCC1 12514,C1(C2CCN(C(c3ccsc3Cl)=O)C2)(NC(=O)Cc2ccc(F)cc2)CC1 12515,CC(C)CC(CNC(C1CC1OC(C)(C)C)=O)C(=O)NCc1cscc1Cl 12516,C1(N(C(c2cc(CCC)on2)=O)C)CCCN(C(=O)CC2C(CC)C2(F)F)C1 12517,c1(C(N(CCNC(Cc2cnc(C)s2)=O)C)=O)cc(F)c(C)cc1O 12518,C1(C)(C(N2CCC(CCNC(C3(C(=O)NC)CCC3)=O)C2)=O)CCCCO1 12519,N1(C(CSCCOC)=O)CCC2(CC(C(=O)N(C)Cc3ccc(F)cc3)C2)C1 12520,N1(C(C2C(C)CC2)=O)CCC(C(C)(O)CNC(c2nn(C)cc2Br)=O)CC1 12521,c1(OC)c(C)cc(C(=O)N(CC)CC2CCCN2C(=O)C(O)P(C)(C)=O)cc1C 12522,CC1CCc2nc(Cl)nc(N3CCCCC(NC(c4coc(Cl)c4)=O)C3)c2C1 12523,N1(C(C2N(C(C)=O)CSC2)=O)CCC12CN(C(C1CCC1(C)C)=O)C2 12524,C1(CC)CN(C)CCCN1C(C1COCC1NC(=O)C(F)C(C)(F)F)=O 12525,CC(C)CC(=O)NC(c1nocc1C(=O)NCC1CCN1C(C)(C)C)C 12526,Cc1cc(C(=O)N(C(=O)C2=CCCC2)C(C)(C)C)n2ncc(C(=O)O)c2n1.C(C#N)N 12527,C1(C(N(C)CC2CC(F)C2)=O)CC2C=CC1N(C(C1CC=CC1)=O)C2 12528,C1(C(N(CCNC(=O)CSC2CC2)CC)=O)CCn2ncnc2C1 12529,N1(C(CC2NC3CCC2C3)=O)CCCC2(CCC2)C1.CC1=C(C=O)CCC1 12530,c1(SC)c(C(=O)NC2CCC(NC(=O)C(N3CCCCCC3)C)C2)cccc1F 12531,c1(C(N2CCC(CCNC(c3conc3C3CCCO3)=O)C2)C)ccccc1Cl 12532,C(=O)(C1CCc2snnc21)NCC1(CO)CCN(C(Cc2cnc(C)[nH]2)=O)C1 12533,N1(C(C(C)N(C(=O)C=Cc2cn(C)nn2)C)=O)CCCC(C)(N(C)C)C1 12534,N1(C(CCS(=O)(=O)NC)=O)CC2(C1)CN(C(C1CCC3(CC1)CC3)=O)CCO2 12535,C1(NC(C2C3COCC23)=O)CN(C(=O)C=CCF)C2(CCC2)C1 12536,c1(CCNC(C=C(CNC(CCCOC)=O)C)=O)cccc(C)n1 12537,C1(NC(Cc2ncc(CC)[nH]2)=O)CN(C(=O)Cn2cnccc2=O)CC1CC 12538,c1(OC)c(Cl)cc(C(=O)N(CCC(C)NC(c2cc(C)oc2C)=O)C)cc1Cl 12539,N1(C(C(c2ccc(OC)cc2)CC)=O)CC(NC(c2occc2C)=O)CC(C)C1 12540,C(=O)(C(C)(C)C)NCC(CC)NC(=O)C=Cc1ccco1.C(=O)(CC)N 12541,c1(CS(=O)(=O)NC(c2nc(-c3ccncc3)cs2)C)ccc(S(C)=O)cc1 12542,CC1CC(NC(c2cc(N)ccc2Cl)=O)CCN1C(=O)C=Cc1ncc[nH]1 12543,C(c1ccc(C)c(C)c1)=CC(N1CCC(NC(C2C(C=C)CC2)=O)C(F)C1)=O 12544,N1(CC(=O)NCC2(C(=O)NC(C(O)CO)C3CC3)CCCO2)CCCNC1=O 12545,c1(C(=O)NCCN(c2csc(C)c2)C2(CC)CC2)ccc([N+](=O)[O-])c(C(F)(F)F)c1 12546,CC(CCc1ccncc1)N=c1[nH]c2c(c(=NCCCCOC)[nH]1)COC2 12547,N1(C(C=CCOC)=O)CCC(C)C(NC(c2cc(OC)n(C)n2)=O)C1C 12548,CCCCCCCCC(=O)NC1CC1NC(c1ccc(C(N)=O)s1)=O 12549,C(=O)(C1=C(Cl)CCOC1)N1CC(N(C(=O)C(F)=CCCF)C)C(O)C1 12550,N1(C(CC(C)O)=O)CC(CNC(=O)CC2C=CCC2)C(F)(CO)C1 12551,C1(NC(CN(C)C(N)=O)=O)C2CCC1N(C(=O)Cc1cncc(F)c1)C2 12552,N1(C(c2c(C)noc2)=O)CCC2OCCN(C(c3cc4cccn4cn3)=O)C2C1 12553,n1(CCCC)nnnc1C(c1ccncc1)NCCSCC1CCCC1 12554,N1(C(c2c(CCC)n[nH]c2)=O)CC(CNC(c2ccn(CCF)n2)=O)CC1(C)C 12555,c1(NC(C(C2CCN(Cc3ccsc3)CC2)C)=O)cc(Cl)ccn1 12556,N1(C(Cc2cnn(C)n2)=O)CCC(CNC(=O)COCCO)C(F)(F)CC1 12557,N1(C(CC2CC(C)N(C(=O)CC(C)(C)C3CC3)C2)=O)CC2C3CCC(O3)C2C1 12558,c1(OC(C)C(=O)NC(C)CC2CN(C(C3CSCN3C)=O)C2)ccc(F)nc1 12559,N1(C(c2cc(C)oc2C)=O)CCC(NC(=O)Cc2cc[nH]n2)C(CO)CC1 12560,c1(C(=O)NCC2CC(NC(=O)CSc3ccccn3)C2)cc2ccccc2o1 12561,C1(C(N(C)Cc2c(CNC(CSC)=O)cccc2)=O)CCOCC1(C)C 12562,C1(NC(c2cc(C)ncc2C)=O)CC2CN(C(C34CC(CO)(C3)C4)=O)CC2C1 12563,c1(NC2C3CN(C(C4CC=C(C)CC4)=O)CC32)nc2cc(C)ccc2o1 12564,CC(CO)C(=O)NCCSCC(=O)NC1(c2nc[nH]n2)CCC1 12565,C1(OC)CC(NC(=O)C=CBr)CN(C(=O)CC2CCSCC2)C1 12566,C(=O)(CCCC(=O)NC(=O)C=Cc1ccsc1)NC1C(CC(=O)OCC)CCC1 12567,Cc1ccc(C(N2CCC(CF)(NC(c3sc(C)c(C)c3C)=O)C2)=O)c(Cl)c1C 12568,CC1(C(=O)NCC2CC(NC(c3cccc(CF)c3)=O)C2)CC2CC2C1 12569,Cc1ccc(C(=O)NC(C)CCNC(=O)C(C)(C)c2nccs2)s1 12570,N1(C(CCc2c(C)cccn2)=O)CCC(CNC(C2CCCOC2)=O)C(C)C1 12571,C=CCC(CC(C)C)C(=O)N(CC(O)CNC(=O)COc1ccc(F)c(F)c1)C 12572,C#Cc1ccc(C(=O)NC2CCC(NC(=O)Cc3cn(C)nc3C)C2)nc1 12573,N1(C(C(CN(C)C)N(C)C)=O)CCCC(CC(=O)NCC2CC(C)(C)CO2)CC1 12574,C(C1=NOC2C3CCC(C3)C12)N(C1CC(C2CCCC2)C1)Cc1c(Cl)cccn1 12575,CC1CN(C(c2ccncc2)=O)CC(CCNC(=O)Cn2ncccc2=O)O1 12576,C(=O)(C(C)(C)C(C)(F)F)NCC1N(C(CC(CC)SC)=O)CCOC1 12577,c1(C(=O)NCC#CCNC(c2cc(CC)nnc2C)=O)cnc2ccnn2c1C 12578,N1(C(c2ccc(C)nc2C2CC2)=O)CCOC2(CCN(CC3CCC3)CC2)C1 12579,C1(C(=O)NC2CC(CNC(C3CC4(CCC4)C3)=O)C2)CC12CCCOC2 12580,C1(NC(C2CC=CCC2)=O)CC2CC1CN(C(=O)C=C1CCOCC1)C2 12581,CC1(C#N)CCN(C(=O)C(C2(O)CN(C(c3c[nH][nH]c3=N)=O)C2)F)C1 12582,N1(C(=O)OC(C)(C)C)CCCCCC1N=c1ccc(Br)n[nH]1 12583,CC1CN(C(=O)Cc2nc(C3CC3)n[nH]2)CC1NC(=O)CC1CC1 12584,CON1CCC(C(=O)NC(C)(C)CNC(=O)CSC2CCCCO2)CC1 12585,C1(C(=O)NC2CC3(C(NC(c4c(C)nc(CO)s4)=O)C3)C2)COC2CCCCC12 12586,C(=O)(C(C)(C)C(C)O)NCCn1cc(C(N(CCCC)CCOC)=O)nn1 12587,c1(COC(C)C)ccc(C(=O)NCC2(C)CCCN2C(C2CC(C)=NO2)=O)cc1 12588,N1(C(C(CC2CCCC2)NC(CCCSC)=O)=O)CC2CCC(C1)C2C#N 12589,C#CCC(C(=O)NCCCSC)NC(=O)C(=Cc1cn[nH]c1)C 12590,C1(SC)CCN(C(=O)CCOCCN(C(=O)C(C)Cc2cnc[nH]2)C)C1 12591,CN1CCN(C(c2sccc2CN)=O)C(CO)C1.C1(N2CC(=O)N2C)CCCC1 12592,C(=O)(C(C)S(=O)(=O)C(C)C)NCC(CN(C(C(CC)(CC)CC)=O)C)C 12593,C1(c2nnnn2CCc2ccccc2)(NCC2(COC)CC2)CCCSC1 12594,c1(CC(=O)N(C(C)CNC(c2cnccc2Cl)=O)CC)ccc(OC)c(C)c1 12595,C1(C)(N(C)C)CCCN(C(=O)COCCNC(=O)Cc2ccnn2C)C1 12596,N1(C(C2N(C(CC(C)=C(C)C)=O)C(C)CC2)=O)C2CCC1COC2 12597,CC1CCCC(CC(=O)NC2CCCC(C(=O)Nc3cccc(F)c3)C2)O1 12598,c1(C(=O)NC2C(NC(c3c(C)cco3)=O)CC2)cc(F)c(F)c(O)c1F 12599,c1(C(=O)NC(C(=O)NCc2c(C)scn2)C2CC2)cnc(C)n1C 12600,CCCCC(S(=O)(=O)NC(=O)C(c1ccc(Br)nc1)(C)C)c1ccccc1 12601,CC(C)CC(C)(CNC(c1cc(Br)n[nH]1)=O)NC(c1ccc(Cl)o1)=O 12602,C=C(C)C1OCCC1C(N1CCC(CO)(CNC(c2cncc(CC)c2)=O)C1)=O 12603,N1(C(CSC)=O)CCCC(NC(=O)CC(C)CC)(OC(=O)NCCOC(C)(C)C)C1 12604,N#Cc1ccc(NC(CNC(c2ccc(C3CC3)cc2)=O)C2CC2)c([N+](=O)[O-])c1 12605,c1(C(N2CCN(C(C34CC(C)(C3)C4)=O)C3C2C3)=O)nncc2c1CCCC2 12606,N1(C(c2c(CC)ncs2)=O)C2CCC1CN(C(=O)Cc1csc(=N)[nH]1)C2 12607,c1(CNC(CC=C)=O)nc2c(s1)CCN(C(=O)CS(=O)(=O)N1CCOCC1)C2 12608,C1(F)(C(=O)NCC2CC(NC(Cc3cnc(C)o3)=O)C2)CCCOC1 12609,C(CCC(=O)N(C1CCC(NC(=O)C(C)(O)C2CCCCC2)C1)C)N(C(C)=O)C 12610,c1(OC)nc(Cl)ccc1C(N1CCC(NC(c2ncccc2C)=O)CC1C)=O 12611,N1(C(CCCn2cc(CC(C)(C)CO)nn2)=O)CC2CC2(CN2CCCC2)C1 12612,CCCCCC(CC)C(=O)NCc1c[nH]nc1C(=O)N(CC(=O)OC)CC1CC1 12613,N1(C(c2cc(OCC)n[nH]2)=O)CCC2(C(=O)NC(C3CCOC3)C)CC2C1 12614,N1(CC(=O)NC2C3CC2N(C(c2snc(O)c2Cl)=O)C3)CCCCCCC1=O 12615,c1(C2(CNC(F)CF)CCCC2)ccc(Cl)cc1 12616,C=C(C)C(C)(C)C(=O)NC1COCC1NC(=O)CCC(=O)c1ccncc1 12617,N1(C(C(CC)N(CC)CC)=O)C2CCC1CC(NC(=O)CC1CC(F)C1)C2 12618,C(=O)(N1CCCc2nncn21)C1C2(CCN(C(c3cc(OCC)no3)=O)C2)C1 12619,Cc1nc(-c2ccccn2)[nH]c(=NC(C)CN(C(=O)CCCCCO)C)c1C 12620,C(N=c1nc2c(c[nH]1)COCC2)C1CCCC(NC(c2ccc(C)c(F)n2)=O)C1 12621,C1(NC(C(=C(C)C2CC2)F)=O)CN(C(C23CCCC(C2)OC3)=O)C2CCCCC12 12622,C(CCS(=O)(=O)c1ccc(F)cc1)N(CCCNC(C1CC2CCC1O2)=O)C 12623,c1(CC(=O)N(C2CC(NC(c3cccs3)=O)C2)C)cccc(N2CCCCC2)c1 12624,C=CCC(C)(C)C(=O)NCC(C)(C1CC1)NC(c1ccnc(S)c1)=O 12625,C1(NC(C=CSC)=O)CS(=O)(=O)C2CN(C(c3cc(Cl)no3)=O)CC12 12626,Cc1nn(CC(=O)NC2CCCC2CNC(c2cncc(N)n2)=O)cc1[N+](=O)[O-] 12627,C1(C(N2CCC(O)(C(C)NC(=O)COCCF)C2)=O)CS(=O)(=O)CC(=O)N1 12628,c1(NCC2C(C)CCN(C(=O)C(C)CC3CCCC3)C2)ncnc2cnccc12 12629,C1(C(=O)NCCN(C)C(c2ccc3c(c2)OCC3)=O)C2C3CC4C1C1C2CC3C41 12630,N1(C(c2c(C)cnnc2)=O)CCC2(CC2)CC1C(=O)NCc1ncn(C2CC2)n1 12631,C1(C)(CNC(c2c(CC)noc2C)=O)CN(C(C2(C)CCCC2(F)F)=O)CC1C 12632,N1(C(c2ccn(CC)c2C)=O)CC2(C1)CN(C(c1cc(C(F)F)[nH]n1)=O)C2 12633,C(=O)(C(F)(F)CCC)N1C(C(=O)NCCCCC#C)CSC1 12634,CC(CC(F)(F)F)C(=O)N1CC2(CC2)CC1CNC(=O)CC12CCCC1C2 12635,C1(C)(C(=O)NC(CCOC)C(=O)NCc2cc(C)nc(O)c2)CCCN(C)C1 12636,c1(C(N2CC3(N(c4nccc(C#N)n4)CC3)C2)=O)cccc2c1OC(F)(F)O2 12637,Cc1csc(C(=O)N(C)CCOCCNC(=O)C(N2CCN(C)CC2)C)c1Cl 12638,c1(C(=O)OC(C)C(=O)N2CC(CC3CC3)C2)cc(Br)cs1 12639,N1(C(CCSC)=O)CCCC2(NC(c3ccc(CN(C)C)cc3)=O)CC12 12640,N1(C(C2(C3N(C(c4cc(C(C)C)[nH]n4)=O)CCC3)CC2)=O)CCC(C)(C#N)CC1 12641,C1(CCNC(C(C)OC)=O)CCCN(C(c2cnc(C3CC3)[nH]2)=O)C1 12642,c1(NC(C2(C)CCCN(C(C(C)OC)=O)C2)=O)cc2ccccc2cc1O 12643,C12(CNC(=O)NC3CC(C)(C#N)C3)CCC(N=[N+]=[N-])(CC1)C2 12644,C1(C(N)=O)CC12CCN(Cc1cc(OCC(=O)O)c(O)c(OC)c1)CC2 12645,Cc1ccn2ncc(C(N3CCN(C(=O)CNC=O)CC(CO)C3)=O)c2n1 12646,N=c1[nH]c2c(s1)CCCC2C(=O)NCC1(O)CCCN(C(=O)C(O)C(F)(F)F)C1 12647,CC(C)(CCCO)NC(C1CSCCN1C(C1CC(=O)C1(C)C)=O)=O 12648,c1(C(=O)NCCN(CCC)C(c2c[nH]nc2S(N)(=O)=O)=O)cc2n(n1)CCOC2 12649,C1(C(=O)NC2(CC(=O)N(CC(C)N(C(C)=O)C)C)CC2)CCCC(F)C1 12650,c1(C(=O)NC2CC(N(C)C)C2)ccnc(CNC(C2(N3CCCC3)CCC2)=O)c1 12651,c1(NC(CC)=O)cncc(C(N2CC=CC2CNC(=O)C=C2CCC2)=O)c1 12652,CN1CC(C(=O)NCCCC2CCCN(C(c3ccccn3)=O)C2)CC1=O 12653,C12(NC(C3OCCN(C(C)C)C3)=O)CC(CNC(=O)C(C)C(F)F)(C1)OC2C 12654,N1(C(C(C)OCCCC)=O)CC2C(CNC(=O)CNS(=O)(=O)NC)C2C1 12655,C1(NC(=O)C(N2CCOC(C3CC3)CC2)=O)CCC2(CCOCC2)C1 12656,C(=O)(CC1=CCOCC1)NC(COC)CC(=O)N1CC(OCCSC)C1 12657,C(C(=O)NCCC1(C)CCOC1)(C(C)(C)O)NC(C1CCC(CC)O1)=O 12658,c1(C(=O)NC(CN(C(=O)CCCc2ccc(C)s2)CC)C)cc(CC(C)C)on1 12659,CCCCCCCC1CCC1.C(=O)(CCCn1cc(C(C)(C)CO)nn1)N=C=O 12660,C1(NC(COC2(C)CCCC2)=O)CCN(C(C2CN(C3CCC3)C2)=O)C1C(=O)O 12661,N12CC(C(n3ccnn3)C1)C2=O.CC1C(NC(=O)CSc2cccnc2)C1(F)F 12662,C1(C(=O)NCc2n(C(C)C)ncn2)CCN(c2nc(C(C)(C)C)co2)CC1 12663,C(C(O)CC(=O)NCC(=O)NC(C)C)NC(c1c(COC)cc[nH]1)=O 12664,O=C1CCC(C(=O)NCCOC2CN(C(c3ccccc3C(F)F)=O)C2)CN1 12665,c1(CC(N2CCC(CC=C)(NC(=O)Cn3nccc3C)C2)=O)cccc(C)c1Cl 12666,Cc1cc(C(N2CC3C(NC(=O)C(O)Cn4cncn4)C3C2)=O)sc1C 12667,N1(c2c(Br)ccc(C(C)C)n2)CCN(C(C(C)(C)C)=O)CC(C)(C)C1 12668,c1(C(N(C2CN(C(c3cnc(CCC)s3)=O)CC2O)C)=O)nccc2ccsc12 12669,Cc1cc(Cl)c(NC(c2cc(F)c(Cl)cc2O)=O)cc1O 12670,CC(C)(C#CC(=O)NCC(C)(O)C1CC1)CNC(=O)CN1CCOC1=O 12671,C1(C(=O)NCc2cn(CC(=O)NC3(C(=O)OCC)CC3)nn2)CCCCC1F 12672,CC1COc2ccc(C(N3CC4CN(C(=O)CC5=CCCC5)CC4(C)C3)=O)cc21 12673,N#Cc1cn[nH]c1C(=O)NCCC1CCN(C(C2C(Cl)(Cl)C23CC3)=O)C1 12674,C(=O)(CCCCCC(C)O)N(CCOCCCNC(C(C)OC(C)=O)=O)C 12675,Cc1cc(Cl)c(Cl)cc1C(=O)OCc1ncoc1C(C)C 12676,C(N=c1[nH]c(NC2CCCn3ncnc32)nc2ccccc12)c1cc(C)nn1C 12677,S1(=O)(=O)c2cnccc2N(Cc2ccc(Cl)cc2)C1.C(C(C)C#N)N(CC)CC 12678,c1(C2C(CNC(=O)Nc3sncc3Br)CC2)ccccc1 12679,N1(C(CCCCCN(C)C)=O)CC2CCC1C(NC(c1cncnc1)=O)C2 12680,c1(C(=O)NC2(CC=C)CCN(C(=O)CC(C)OC)C2)cc(C)cc(Br)c1 12681,C1(C(N(C)CC2(O)CN(C(=O)C=Cc3cc[nH]n3)C2)=O)COCCN1C 12682,c1(C(N(CC(CC)NC(=O)CCC2CC=C(C)CC2)CC)=O)cccc(C)c1F 12683,N1(C(C(c2ccn(C)c2)C)=O)CC2CCCC(N(C(=O)CN(C)CCO)C)C2C1 12684,c1(NC(C)=O)c[nH]c(C)c1C(=O)NCC=C1CCN(C(=O)C=C2CC2)CC1 12685,CN1CCCC2CN(c3cc(C(=O)O)c4c(c3)CCS4)CCC12 12686,CCN=c1[nH]cc(C(=O)NCC(Cn2cc(CC3CCCC3)nn2)OC)s1 12687,N1(C(CCn2ccc(C)n2)=O)CCC(C)N(C(=O)CC2COCC2O)CC1 12688,C(=O)(C1=C(Cl)CCOC1)N1CCCC(C)C1CN=c1[nH]nc(C(F)F)o1 12689,N1(C(C(C)(C)SC)=O)CCN(C(c2n[nH]c3c2CCC3)=O)C(C2CCC2)C1 12690,c1(CNC(C(C)NC(=O)CCCc2cnn[nH]2)=O)c(O)cccc1F 12691,c1(C(=O)NC(C)CNC(=O)Cc2ccc(N)cc2)cc2ccc(O)nc2s1 12692,N1(C(c2cccc(N)n2)=O)CCOCC(F)(CNC(C2(Cl)CC2(F)F)=O)C1 12693,CCC(CN=c1cc(NCCN2CCCCC2C)nc[nH]1)OC 12694,CC#CCCC(=O)NCC(C1CCOC1)NC(=O)Cc1cnn(C)c1C(F)F 12695,C1(C(=O)NC2COCCC2O)COC2(C1)CN(C(C1CC1(Cl)Cl)=O)C2 12696,c1(C(N2CC(OC)C(C(=O)NC3CCCC3CF)C2)=O)cc2n(n1)CCO2 12697,CC(C)CCC(C(=O)NCC(C)(O)CO)NC(c1cn(C)cn1)=O 12698,c1(NC(CC)=O)ccc(C)c(C(=O)NCc2ncc(Br)cc2N)c1 12699,C1(NC(=O)C=CC2CCOC2)CCCC12CCN(C(C13CC(C1)C3)=O)CC2 12700,c1(CCC(=O)NCC(C)(CO)NC(C2(OC(C)=O)CC2)=O)nnc(S)n1C 12701,N1(C(c2ccc(OC)c(O)c2)=O)CCC2(C1)CN(C(c1ncsc1C1CC1)=O)C2 12702,c1(C(N2CCN(C(C3CC(=C)C3)=O)C(C)C2)=O)cc2ccccc2nc1O 12703,c1(NC2CC(CNC(CCC(=O)N(CC)CC)=O)C2)ncn(C)c(=O)c1Br 12704,Cc1cnn2ccc(C(N3CCC(C(C)NC(=O)CP(C)(C)=O)C3)=O)nc12 12705,C1(CC)CN(C(c2cc(C)ccc2Cl)C(=O)NC2CCCC2)C2(CCC2)C1 12706,N1(C(CCP(C)(C)=O)=O)CCC(C2(NC(=O)Cn3ccc(O)nc3=O)CC2)C1 12707,C(=O)(C(O)P(C)(C)=O)NCC(CN(C)C(c1cncc(C(C)(C)C)c1)=O)(C)C 12708,N1(C(c2ccc(OC)s2)=O)CC(CO)C2(C1)CN(C(C1(C#N)CCSCC1)=O)C2 12709,C(=O)(C(CNC(=O)CC(F)(F)F)C(C)(C)C)NCCc1cn(CC)nn1 12710,CC(C)S(=O)(=O)c1cccc(C(=O)NC(C)CN(C)C(C2COCCO2)=O)c1 12711,c1(C(=O)NC23CC(CNC(CC4CCCN(C)C4)=O)(C2)C3)ccc(F)cc1Cl 12712,C(=O)(C(F)(CNC(=O)OCc1ccccc1)C(C)C)Nc1c(OC)ncc(C)c1 12713,Cn1cc(-c2n[nH]c(CNCc3ccccn3)n2)cn1 12714,C(CCCCC(C(=O)NC(C)(C)C)N1CCn2nc(C)c(I)c2C1)OC 12715,O=S(=O)(c1ccccc1N1CCCCC1)NCCC1CCC1OCc1ccccc1 12716,C(=O)(CCCC(F)(F)F)N1CCC(C)C(NC(=O)C(c2ccccc2F)(F)F)C1 12717,C1(C(C)C)CN(C(=O)Cn2nc(O)ccc2=O)CCN1C(c1cc(=O)cc[nH]1)=O 12718,c1(C(N(CC(C)CNC(=O)C(O)C2CCC2)C)=O)cccc(S(=O)(=O)CF)c1 12719,C12(C(=O)NC3CCN(C(Cc4cn(CC)nc4)=O)CC3O)CC1Cc1c[nH]nc12 12720,C(N=c1[nH]c(=NC)[nH]c(=NCC2C=CCCC2)[nH]1)c1ccc(N(CC)CC)cc1 12721,c1(N(C)CCOC(F)F)nc(=NCc2cc(Br)ccc2C)[nH]c2c1CSC2 12722,Cn1cc(C=CC(=O)NCC2(C(=O)NCC3CC3C3CC3)CCC2)nn1 12723,C1(C(C)NC(C(CC)NC(N)=O)=O)CCN(C(=O)CCCC2CC2)CC1 12724,C1(COC)(CNC(=O)CCC2CCOCC2)CCN(C(C2CC(=O)N(C)C2)=O)C1 12725,C#CCC(C)(C)C(=O)NC(CNC(=O)C(C)n1ccnc1)CCOC 12726,C1(NC(C(=O)N(C)C)=O)CC(CNC(=O)CCC(=O)c2cccc(N)c2)C1(C)C 12727,C=C(F)CN=c1[nH]c(N2CCN(c3nsc(C4CC4)n3)CC2)nc2c1COC2 12728,N1(C(C(C2(O)CN(C(C(C)OC(C)=O)=O)C2)F)=O)CCc2ncn(C)c2C1 12729,c1(C(=O)OCC)c(NC(=O)CCCc2ccsc2)sc2c1CCC(C)C2 12730,C(=O)(C(C(F)(F)F)C(F)(F)F)NCC(N1CC(C)(C)c2c1cccc2)=O 12731,C(=O)(C(C)(C)C(O)C(C)C)NC1CC=C(C(=O)N2C(C)CC(C)C2)C1.CC(=O)N 12732,S(=O)(=O)(c1ccncc1)NC(c1ccco1)=O.c12ccccc1N2C(C)=O 12733,C1(NC(c2cnoc2C2CC2)=O)COCCC1NC(C1CC1C(F)(F)F)=O 12734,CCC(C(=O)NC(CNC(c1cc(C2CC2)ns1)=O)Cc1ccccc1)NC(N)=O 12735,C1(C2CN(C(=O)C(F)C3CC3)C2)(NC(C(c2ccc(C#N)cc2)C)=O)CC1 12736,c1(C(N2CCC(C)C2CNC(=O)CCn2ncn(C)c2=O)=O)ncc(N)cc1Cl 12737,c1(C(N(C(c2ccccc2)CNC(=O)C(C)C2(O)CCC2)C)=O)cccnc1O 12738,c1(C(=O)OCC)nc(CN(C(C2CCC(C(C)C)CC2)=O)CCOC)n(C)n1 12739,C1(NC(C2C(C)N(C)CC2)=O)CCC12CN(C(=O)CCc1ccc(CO)cc1)C2 12740,C(CC(=O)N=c1cc[nH]c2ccsc12)NC(=O)OCC 12741,C1(CCNC(c2cnn(CCC)c2C)=O)CCN(C(=O)CN(C)CCO)C(C)C1 12742,C1(C(N2C(C)CC(NC(C3CC3C3CC3)=O)CC2)=O)CCCCC1N=[N+]=[N-] 12743,CCCC(C)(C)CC(=O)N1CC2CCC2(CC(=O)NCc2cc(C)ncn2)C1 12744,c1(C(N(C(C)C(=O)NC(C)CN2CCCC2=O)C2CC2)=O)cc(=O)cc[nH]1 12745,CN=c1ncc(-c2nc(C(N3CC4CCC(C3)O4)=O)cs2)c[nH]1 12746,C1(NC(c2cnn(-c3nccs3)c2)=O)CN(C(c2ccsc2)=O)CCC1CO 12747,N1(C(Cc2scc(C)c2)=O)CCC(C)(NC(c2coc(C(F)(F)F)c2)=O)C1 12748,C1(NC(CCCN(C(C)C)C)=O)CCC(CNC(C2CC(CN(C)C)C2)=O)CC1 12749,N1(C(=O)C(=O)NC2CCC=CCCC2)CCc2cc(C3CCCCC3)ccc2C1 12750,C(=O)(CC(O)CC(C)C)NCC(CCC)C(=O)NC1C=CC(C(=O)OC)C1 12751,C(=O)(C1c2c[nH]nc2CN1C(=O)CCCn1ccnc1)NCC(N1CCCC1)C 12752,c1(C(=O)NCCOCCC(=O)NCC=C)ccc(CC)o1 12753,c1(NC(C)=O)ccc(Cl)c(C(=O)NCC(C)NC(=O)C(c2ccccc2Cl)O)c1 12754,c1(CC)cc(C(=O)NCc2n[nH]cc2C(=O)NC2CCCC2C#N)ncn1 12755,c1(C(N2CCCCC2C(=O)Nc2csc(Br)c2)=O)cc(F)cc(Br)c1Cl 12756,C(=O)(C1=CCC(NC(=O)CCC2(C#N)CCC2)C1)NCC(=O)NCCC 12757,C1(C(=O)NCCNCC2CCC(C(=O)OC)C2)CCCC(C)(C)CC1 12758,N1(C(C(CCC)O)=O)CCC(C(F)(F)F)CC1CNC(c1nncn1C1CC1)=O 12759,Cn1ccn2ncc(C(N3CC4C(NC(=O)C=Cc5cc[nH]c5)C4C3)=O)c12 12760,C1(NC(C(CSC)O)=O)CC2CC1CC2C(=O)NC(CCO)C(C)(C)C 12761,C=CC(CC)CC(=O)Nc1c[nH]c(=N)c(C)c1.C12CN(CC1C=C)C2=O 12762,c1(C(N2C(C)CC(CNC(=O)C=Cc3cc[nH]c3)C2)=O)cnc2n1CCS2 12763,Cc1nn(C)c2ncc(C(=O)NCCCC(C)NC(c3nc(=O)n(C)[nH]3)=O)cc12 12764,C(=O)(C1Cc2ccc(Cl)cc21)NC(CCCC)CNC(c1cc(C2CC2)[nH]n1)=O 12765,C(=O)(C(C)(C)C1CCCO1)N(CCCN(C(=O)Cc1cccnc1)C)C 12766,c1(C(N2C(C)(CNC(c3ccsc3C(F)F)=O)CCC2)=O)ccc2nonc2c1 12767,c1(CCC(=O)NC(C)CNC(C2(CC3CCC3)CC2)=O)ccc(Br)s1 12768,C(=O)(C1=CCCC1P(C)(C)=O)N1CC(C)C(CNC(=O)C(C)(C)CN(C)C)C1 12769,c1(C(C)NC(=O)N(C)Cc2cc(Cl)ccn2)ccc(Br)cc1Cl 12770,C(=O)(C(CNC(=O)CC1CCOC1)N(C)C)N1CC(OC)C1 12771,N1(C(C2(CC)COC2)=O)CCC2(CC1)CC2C(=O)NOCC(O)CO 12772,c1(C(=O)NCC2CCC(NC(c3c(CC)non3)=O)C2)nccc2c1NCCC2 12773,N1(C(c2cc(Br)cs2)=O)CCOC(CNS(=O)(=O)CCBr)C1 12774,C(=O)(C1=Cc2ccccc2C1O)N1CCC(CNC(c2cncc(SC)c2)=O)C1 12775,CC1(C(=O)NCCN(C(=O)CSC2CC2)Cc2ccccc2Cl)COCCO1 12776,C(=O)(C(C)C(F)(F)F)N(CC=CC(=O)N(C)Cc1c(CC)noc1)C 12777,CC1(C)NC(=O)CC1C(=O)NCC1(CNC(C2(C)CC3C=CC2C3)=O)CC1(F)F 12778,CCC(CC)CC(=O)N1CC(O)(CNc2nccc(-c3cnccn3)n2)C1 12779,C#Cc1ccc(C(=O)NC(CCN(C)C)C(=O)NCCc2nnc(C)n2C)cc1 12780,C=C(Br)CC(=O)NC(CO)C(C)NC(=O)C=Cc1cnc[nH]1 12781,c1(OC)cscc1C(=O)NC(CN(C)C)C(=O)NCc1cncnc1 12782,CCCC(CCCNC(C1CC1(F)F)=O)NC(=O)CCCCc1ccccc1 12783,c1(C(=O)NC2CCC(NC(CCSCCCC)=O)C2)nccnc1C(F)(F)F 12784,C1(F)(C(=O)NCCC(=C)CNC(=O)COc2cc(Cl)ccc2C)CCS(=O)(=O)C1 12785,CCCC(CC)CCC(=O)NC(C)CNC(C1CCCCC1OC)=O 12786,CC1=NN(C)C(=O)C1CC(=O)NC12CC1CN(C(=O)CC1CCOCC1)C2 12787,N1(C(CCSCC)=O)CCC(CNC(=O)C(O)Cc2ccccn2)(OC)C1 12788,C12COCCN1C(=O)CNC2.C1(CN(C(C(=O)N(C)C)=O)C)CCCCO1 12789,C1(CN(C(=O)C(O)Cn2cncn2)C)CCCCN1C(=O)CCC#N 12790,c1(C(=O)NCCN2CCCN(C(C3C(OC)C3)=O)CC2)cccc2c1ncn2C 12791,Cc1cccnc1CCC(=O)NC1CCC1NC(c1ccc(CO)cc1)=O 12792,c1(OC)ccc(C(=O)NCc2cc(C(F)(F)F)nn2C)c2cccnc12 12793,C1(O)(CNC(C2C(C)C2C)=O)CCN(C(c2cc(C(F)F)nn2C)=O)C1 12794,C1(C(=O)NCc2ncc(C)nc2)CC12CCN(C(=O)CCc1cncn1C)CC2 12795,C1(NC(C=CCCC)=O)CN(C(=O)C(c2ccc(Cl)cc2)=O)CC1C1CCCO1 12796,CCC(CC(=O)NC1CCN(C(C2CC23CCCCC3)=O)C1(C)C)CC(F)(F)F 12797,c1(C(=O)NC(C)C(C)NC(c2c(F)cncc2Cl)=O)cc(F)cc2cc[nH]c12 12798,C1(CNC(C=COCC)=O)C2CN(C(=O)CC3(C(F)(F)F)CNC(=O)C3)CC12 12799,N1(CC)CCN(CC(=O)NCC(CO)NC(=O)CN(c2ccco2)C)CC1 12800,N1(C(CCN(C(CCOCCC)=O)C)=O)CCC2CC2C1 12801,c1(-c2c(CNC(CCC(=O)OC)=O)cccc2)cnc(C)c(C)c1 12802,C(=O)(C(C)CCC(C)(C)C)N1C(C(=O)Nc2ccc(C)cc2)CC=CC1 12803,c1(N(C)Cc2c(C)ccnc2)nc(N(C)CC2CC(F)C2)nc2ncn(C)c12 12804,c1(C(=O)NC2(C)CC2)cn2c(n1)CCN(C(=O)Cn1cc(S(C)(=O)=O)cn1)CC2 12805,C(=O)(C1=CS(=O)(=O)CCC1)NCC(C)(O)CNC(c1ccncc1C(F)(F)F)=O 12806,C1(C(C)(C)CNC(=O)CNC(N)=O)CCCCN1C(=O)C=Cc1ccco1 12807,C(=O)(CCC(=O)NC1CC(c2ccccc2)(CNC(=O)C=CS(C)=O)C1)NC 12808,Cc1cnc(C)c(C(=O)NCC(C)CN(C)C(c2sc(F)cc2Cl)=O)c1 12809,C(=O)(C1=CC2CCC1C2)N1CCCC(N(C)C(c2cccc(Cl)c2)=O)C1 12810,c1(NC(C2N(C(c3nc(CC)oc3)=O)CCC2)=O)c(C)ccc(I)c1C 12811,c1(N2CCC(C(C)(C)CNC(C3CCCC(O)C3)=O)CC2)nccnc1C#N 12812,C1(NC(C=C(C)Cl)=O)CCCC(NC(c2cccc(N3CCNC3=O)c2)=O)CC1 12813,C1(NC(Cn2c(C)ccc2C)=O)CCN(C(c2ccncc2Br)=O)C12CCC2 12814,c1(N(C)Cc2nccs2)nc2cc[nH]c2c(=NCC2CCc3cccnc32)[nH]1 12815,O=C(C1=C(Cl)CCCC1)N(CC(=O)NCC12CCCCC1C2)C1CC1 12816,C(C)(CCCCNC(=O)C(C)c1ccon1)NC(c1c(C(C)C)occ1)=O 12817,C1(NC(Cc2c(C)noc2Cl)=O)CC1C1CCN(C(c2cncc(O)c2)=O)CC1 12818,C1(O)(CNC(C2(N(C)C)CC2)=O)CCN(C(c2cc(Cl)ccc2F)=O)CC1 12819,c1(C(=O)NC2(CNC(C=C(CC)C)=O)CCOCC2)cccc2oc(C)cc12 12820,CCC(C)(CNC(c1ccc(C(C)=O)[nH]1)=O)C(=O)NCC1CC(=O)N(C)C1=O 12821,CC(CNC(=O)CC(C)CNC(c1cncn1C)=O)C(F)(F)F 12822,C(=O)(C(C)(C)C(F)(F)F)NC1C(NC(c2cccc(SCCCC)c2)=O)CCC1 12823,CCS(=O)(=O)CCNC(C1(CNC(C2CC2(F)Cl)=O)CC(=C)C1)=O 12824,c1(C(N2CC(CCNC(CS(=O)(=O)NC)=O)OCC2)=O)nn(C)c(Cl)c1Cl 12825,c1(CNC(C(CCOC)NC(=O)CSC(F)F)=O)cccc(F)c1F 12826,C1(NC(CC2(NC(C)=O)CCCCC2)=O)CC(F)CN(C(=O)CCS(C)(=O)=O)C1 12827,c1(N(C(=O)Cc2ccc(CO)cc2)CC2(F)CCNC2)ncnc2ccccc12 12828,N1(C(C(C)CN(C)C)=O)CC2CC(NC(=O)C(=Cc3cccnc3)F)CC1C2 12829,c1(C(=O)NCCCN(C(=O)Cn2nnc(=O)[nH]2)C)ccc(CNC(=O)N(C)C)o1 12830,C1(C(=O)NCC2(CC=C)CCCC2)CN(C)CCN1C(c1ccccc1Cl)=O 12831,C1(O)(COC(c2nc(C)n(-c3ncccn3)n2)=O)CCCC(C)(C)CC1 12832,c1(C(=O)NCCN(CCOC)C(C2CCC(C)S2)=O)cc(Cl)cc2c1OCC2 12833,O=C(N=c1cc[nH][nH]1)C1CC(O)CN1Cc1ccc(-c2ccc(Cl)cc2)cc1 12834,C1(NC(CCCCC=C)=O)CN(C(=O)C(CC)N2CCCC2=O)CC(F)(F)C1 12835,N1(C(=O)COc2ccc(Cl)cn2)CCC2CCCN(C(=O)C3=NOCC3)C2C1 12836,c1(C(N2CCC(CNC(CC(CC)C3CCC3)=O)CC2)=O)nnc2ccccn12 12837,C(C(C)N=c1nc(N2CCOCC3(CC3)C2)c2sccc2[nH]1)c1ccc(SC)cc1 12838,N1(C(CCCC(C)NC(CC(C)(C)OC)=O)=O)CCCC12CCOC2=O 12839,N1(C(CCOCCOC)=O)CC(NC(c2nccc(OC)c2F)=O)CC(F)C1 12840,CC1CCCCC1(CNC(c1ccc(=O)n(C)n1)=O)NC(=O)CCNC(=O)CO 12841,C(CN=C(NCc1ccco1)N1CCCC(OC(F)F)C1)C1(OCC)CCCC1 12842,N1(C(CC(CC)C)=O)CC2CCC1(CNC(=O)C#CC(C)(C)C)CC2 12843,N1(C(c2cc(CCOC)on2)=O)CC(C)CN(C(=O)CC2CCSC2)CC1C 12844,C1(NC(C(C)n2cnnn2)=O)(CF)CCN(C(=O)C2=COCC2)C1 12845,C(=O)(C#CC1(C)CCCO1)N(CCCCN(C)C(C1(C)CC1Br)=O)C 12846,c1(C(N(C)CC2CCN(C(Cc3c(C)ccs3)=O)CC2)=O)csc2ccncc12 12847,N1(C(c2cc(CC)oc2C)=O)CC2CCC1CN2C(=O)CCC1CCN(C)C1 12848,Cc1nnc2n1C(C(=O)NCCCCCCNC(c1cnc(C(C)O)s1)=O)CC2 12849,Cn1cc(Cl)c(CCNC(=O)NCc2ccc(OCC(F)(F)F)cn2)n1 12850,CC1(C)CC(C(=O)NC2CC3CCCC3C2)CN(C(=O)CN2CCSCC2)C1 12851,C1(NC(=O)CCCn2cccn2)CS(=O)(=O)CC1NC(C12CCCN1CCC2)=O 12852,N1(C(C(CCSC)NC(C2CN(C)CC(C)O2)=O)=O)CCn2nccc2C1 12853,C(=O)(C(F)CCC(C)(C)C)NCc1c(C(=O)Nc2c(C)csc2)nco1 12854,CC1ON=C(C(=O)N(C)CC2CCCN2C(=O)CSC(F)(F)F)C1C 12855,CCCCCC(O)CC(=O)NC1CCCC1NC(C1(C(N)=O)CC1)=O 12856,C1(C)(CNC(C(CC)Sc2nc(=N)[nH][nH]2)=O)CCN(C(=O)OC(C)(C)C)CC1 12857,CCC(CC)CC(F)C(=O)NCCC1(O)CCN(C(C2OCCC2CC)=O)CC1 12858,c1(C(=O)NCCCN(C(C(n2ncc(C)c2)C)=O)C)ccc(C)c2c1CCC2 12859,N1(C(C(C)Oc2ccccn2)=O)CCN(C(=O)CN(C)C2CC2)C(CCNC)C1 12860,c1(OC)ccc(C(CNC(=O)Cc2nnc(C)n2C)NC(=O)C2=NOCC2)cc1 12861,C1(O)(COC)CN(C(C2CCC2CNC(=O)C(C)n2cccn2)=O)C1 12862,CCC(C(=O)NC(c1ccc(-c2cc(NC)sc2)s1)=O)c1ccccc1 12863,Cn1nc(CC(=O)Nc2cc(-c3ccccc3Br)on2)c2ccccc2c1=O 12864,C1(CN(C(CCOC)=O)C)CCCCN1C(c1sccc1OC)=O 12865,C(C1CCCCCC1)=CC(=O)NCC1(F)CN(C(CCC(=C)Cl)=O)C1 12866,C=CC1CN(C(c2cnc(C)c(CC(C)C)c2)=O)CC1NC(=O)C#CC1CC1 12867,CC(C)CC(CNC(C1CC(C)(C)CN1C)=O)C(=O)Nc1ccc(F)cc1CO 12868,CC1CCCC=C1C(=O)NCC1CCC1NC(c1ccn(C(C)(C)C)c1)=O 12869,c1(C(=O)NCC2N(C(CC(c3scc(C)c3)O)=O)CCC2)c(C)coc1C 12870,C(=O)(C1=NOC(CNC(=O)CCOCC)C1)NCC(=C)F 12871,N1(C(C)C(=O)NCCC2CC(NC(C3(C4CC4)CC3)=O)C2)CCCCC1=O 12872,c1(C(C)C)ccoc1C(=O)NC12CC(NC(=O)C(F)C3CCCC3)(C1)C2 12873,c1(C(C)C)ccc(CNC(=O)N(C)CC2CCCN2Cc2cccnc2)cc1 12874,c1(CC)nc(Cl)c(F)c(=NCCCCNC(=O)C(Cc2ccccc2C)CC)[nH]1 12875,c1(C(N2C(CNC(C3C(C=C)C3)=O)CC(C)(C)C2)=O)ccc2oc(=N)[nH]c2c1 12876,N1(C(C(C2CC(C)(C)C2)OC)=O)CCC2(CCC(NC(=O)CC(F)(F)F)C2)C1 12877,C=CCCC(CC(C)C)C(=O)NCC(C)(C)CN(C)C(C1CCOC(=O)CC1)=O 12878,c1(C(=O)NC(CCCC=C)c2ccccc2)[nH]cc2c1CCCC2 12879,N1(C(Cc2cc(C)nn2C)=O)Cc2ccc(CNC(=O)Cc3cnsc3)cc2C1 12880,c1(C(N2C(CN(C(CN(C)CCO)=O)C)COCC2)=O)cc(O)c2ccoc2c1 12881,C(=O)(C#CC1(C)CC1)NC(C)C(=O)NCC(CNC(=O)C(C)(C)C)(C)C 12882,c1(C(=O)NC2CC3CCC2(NC(c2ccon2)=O)C3)cc2ccccn2c1 12883,c1(C(=O)NCCCNC(CSCC(=O)OC)=O)ccc2c[nH]nc2n1 12884,C1(S(C)(=O)=O)(NC(Cc2c(C(C)C)con2)=O)CC1C(F)(F)F 12885,CC(C)(C)CCCC(=O)NCC1(F)CN(C(=O)CC2CCOC(C(C)(C)C)C2)C1 12886,C1(C(N(C(C)C2CC2)CC)=O)CC2CC2N1C(=O)CCOCC1CC1 12887,N1(CCOC)CCC(N=c2[nH]c(N3CCSC(C(F)(F)F)C3)nc3c2COC3)C1 12888,c1(COC)nn[nH]c1C(=O)NC(C)C(C)NC(=O)CNc1nccs1 12889,c1(CC)cccnc1C(=O)NCC1CC2CC2N1C(=O)C(C1CCOCC1)F 12890,C1(NC(C#CC(C)(C)C)=O)CC(N=c2ccnc(Cl)[nH]2)C1(C)C 12891,c1(C(=O)NCC(CNC(CNC(=O)NC)=O)O)c(Br)nc2n1CCCC2 12892,N1(C(C(C2CCC2)OC)=O)CCN(C(c2ccnn2CCF)=O)C(C(F)F)C1 12893,N1(C(C(C)OCC(C)C)=O)CCC(C2CCN(C(C3CCCCN3C)=O)CC2)C1 12894,C1(CCC(=O)NCC(=O)OC)CCCN(C(=O)CCC(C)OC)C1 12895,N1(C(c2n(CC)nnc2)=O)C2CCC1CC(N(C(=O)CN(C1CCSC1)C)C)C2 12896,c1(C(CNC(C2CCCO2)=O)NC(c2cc(C(N)=O)n[nH]2)=O)ccc(F)cc1 12897,c1(C(N2CCC(CNC(CC)=O)C(C)C2)=O)cnc2c(n1)CCCC2 12898,c1(OCC(=O)NCC(CC)N(C(=O)C(F)C2CCC2)C)ccc(Cl)cc1C 12899,N1(C(CCSCC)=O)CCCC2(CCCCC2NC(=O)CC2(O)CCOCC2)C1 12900,C1(C(=O)NCCOC2CN(C(c3ncsc3C3CC3)=O)C2)CCCC2(CCC2)C1 12901,C1(NC(c2cc(OC)n(C)n2)=O)CCCN(C(C2CN(S(C)(=O)=O)C2)=O)CC1F 12902,CC1C(=O)CC1C(=O)NC(C)(CNC(=O)CCC1(C)CC1(F)F)CO 12903,C(C(C(C)(C)C)NC(=O)CCCN1CCCC1)NC(C1CC(OC)C1)=O 12904,N1(C(C2(C)COCCO2)=O)C2CCC1CN(C(c1ccc(C(F)F)nc1)=O)C2 12905,Cc1cc2c(cc1C)OC(C(N1CC(NC(C3C4CCC3CC4)=O)C1)=O)C2 12906,C1(C(=O)NCC2C3CN(C(COCCCC#C)=O)CC32)CCC(S(N)(=O)=O)CC1 12907,C1(NC(C(C)NC(COCCOCC#C)=O)=O)CCOC12CCCC2 12908,N1(C(C(CCCC)NC(=O)CCn2ccnn2)=O)CCC12CCCCC2 12909,C(=O)(C(CC)CC=C)NC(CCCCNC(c1cc(CCCCC)[nH]n1)=O)C 12910,N1(C(c2n(C)cnn2)C(=O)NCC(F)F)CCOC(c2cn(C)cn2)C1 12911,Cc1cc(C(N2CC(NC(=O)CC(C)CF)C2)=O)cc(N)c1 12912,Cc1cc2ccccc2nc1C(=O)NC1CC(C)(NC(=O)C2=CCS(=O)(=O)C2)C1 12913,c1(CN2C(C)CCC(C(=O)OC)C2)cccc(C#N)c1OC 12914,C1(C(N2CCCC(C(=O)Nc3cnn(CCO)c3)C2)=O)CCCC2(CC2)C1 12915,N1(C(Cc2c(C)nsc2)=O)CCC(F)C(NC(c2ccnc(C(F)(F)F)n2)=O)C1 12916,C#CC1CN(C(c2ccc(SC)cc2)=O)CCN1C(C1Cc2nncn2C1)=O 12917,N1(C(C2CCC(C)(C)C2)=O)CC2(CC(NC(c3ccoc3)=O)CO2)C1 12918,C1(NC(CCC(=O)OC)=O)CC(O)CN(C(=O)C(F)(F)c2cnn(C)c2)C1 12919,N1(C(C(CC)NC(N)=O)=O)CC(CNC(=O)CCCF)C(n2cccn2)C1 12920,c1(C(=O)NCC(C2CCCN(C(c3ccc(Cl)cn3)=O)C2)(C)O)cccc(Cl)c1 12921,C1(C(C(=O)OCCCCCC)CC)CCN(c2ccccc2)CC1 12922,Cn1nc(C(N2CC3CC2C3C(N2CCC(F)(CO)C2)=O)=O)cc1O 12923,N1(C(c2cncc(C#C)c2)=O)CCC2CCCC12CNC(=O)C(C)(C(C)C)OC 12924,CCCC(C)(CC)C(=O)NCC1CC(C(=O)Nc2cccc(C(C)=O)c2)=NO1 12925,C1(CC)CN(C(c2ccncc2OC)=O)CC1NC(=O)C1=CCCS1 12926,CCC(CC(=O)NCC(C)CC(=O)N1CC(C)(CCO)C1)C1CCC1 12927,c1(C(=O)NC2CN(C(C(C(C)C)NC=O)=O)C2)cc2c([nH]1)CCC2 12928,C1(CCCCCC)CCCC1(c1nnnn1C1CCC1)NCC1(C)CC1Br 12929,CC12CN(C(=O)COC3CC3)CC1(C)CN(C(C1Cc3cccc(F)c3O1)=O)C2 12930,c1(OCC)ccc(CNC(=O)NC2CCN(C(=O)C(F)n3cccn3)CC2)cc1 12931,CC(CCCCNC(=O)CCc1cc(Cl)cs1)NC(c1coc(Cl)c1)=O 12932,c1(NC(CCC)CC(F)F)ncccc1S(=O)(=O)NC(CCC)CC(F)(F)F 12933,C(CC(C(C)(C)C)NC(c1ccc(F)c(F)c1)=O)N(C(C1CCN(C)C1=O)=O)C 12934,O=C(C1=CCCN(CCn2ccc3ccccc23)C1)NCCCc1ccncc1 12935,C1(NC(C2CCN(CC)C2)=O)CCC2(CC1)CCN(C(=O)C1=NOCC1)C2 12936,C(=O)(C(O)CC(N)=O)N(C)CC1(O)CN(C(C2(OC)CCC(C)C2)=O)C1 12937,C#Cc1ccc(CCC(N2CC3(NC(=O)COCC=C)CCC2C3)=O)cc1 12938,CC(C)CC(O)C(=O)N1CC(O)CC1CNC(C1C2(CC2)C12CC2)=O 12939,C(=O)(C(CO)C(C)(C)C)N1CC(C(C)(C)O)(CNC(C2CCC(C(N)=O)O2)=O)C1 12940,CC(C)CC(CNC(c1cccc(=O)o1)=O)C(=O)N(C)CC1CC1 12941,C1(CNC(CCc2c(OC)cccc2)=O)CCC(C)N(C(c2cc(C)co2)=O)C1 12942,C(C(=O)N(C)CC1CCCOC1)(C(C)(C)C)NC(c1c(CC)ocn1)=O 12943,CC1=C(C(=O)NC2CN(C(c3nn(C)c(Cl)c3Cl)=O)CC2F)SCCO1 12944,C1(CC(N2CCC(CNC(c3ncn(C)n3)C)C2)=O)CCC(=O)C1C 12945,N1(C(c2ccc(C)c(F)c2)=O)CCN(C(=O)C(C)(O)C(C)C)CC(CO)C1 12946,CCC(O)C(F)(F)C(=O)N1CCOCC(CNC(=O)C(C)(C)O)C1 12947,N1(C(C=C(CC)CC)=O)CCC2CCC12CNC(c1ccc(O)c(Br)c1)=O 12948,c1(C(=O)NC2CCCN(C(c3[nH]cc(CC)c3)=O)C2C)cc2c(s1)CCSC2 12949,C1(NC(CC2N(C(C=C(C)C3CC3)=O)C3C2CCC3)=O)CCc2n[nH]cc2C1 12950,c1(C(=O)NC2(c3ccncc3)CC2)cc(Cl)ns1 12951,C1(Br)(C(=O)NCC(CN(C(=O)C2=CC(C)(C)C2)CC)(C)C)C(C)(C)C1(C)C 12952,C(CN=[N+]=[N-])(C(=O)N1CC(OC)C1)NC(C1CCN(CC)C1)=O 12953,C1(C(=O)NCC(O)CC2CCCC2)CC2CC2N1C(C1CCCCO1)=O 12954,Cn1nc2c(c1C(N1CC(NC(=O)CSC(C)(C)C)C3(CC3)C1)=O)COCC2 12955,C(=O)(CC(C)(C)C(F)F)N1CCC(C(C)C(N2CC(CO)C(O)C2)=O)C1 12956,c1(C(N(CCCNC(C2CC2Cl)=O)CC)=O)cc2cc(C)ccc2o1 12957,C1(CNC(C(=Cc2cccs2)C)=O)C2CCC(C2)N1C(=O)CNS(N)(=O)=O 12958,C12(NC(C(CC)C)=O)CCC(n3cc(C=CC(C)C)nn3)(CC1)C2 12959,N1(C(C(C)NC(COC)=O)=O)CCC(CO)(NC(=O)CN2CC=CC2)CC1 12960,n1(CC(=O)NCCCN(C(c2cc(C(=O)OC)no2)=O)CC)cc(Cl)cn1 12961,Cc1[nH]nc(C(N2CCC(n3cc(-c4ccc(CO)cc4)nn3)CC2)=O)c1O 12962,C#CCC(C(=O)NCC(O)CSCC=C)NC(=O)COCC 12963,c1(C(=O)NCC(C)(CO)NC(=O)CSC2CC2)cccc(OC(F)F)c1 12964,N1(C(C2OCCC(NC(c3ccc(C)n3C)=O)C2)=O)CCOC(C)(C)CC1 12965,Cc1cc(=NCc2cnc(C)c(Br)c2)[nH]cc1S(=O)(=O)N(C(C)CN(C)C)C 12966,c1(C(N2CCN(C(c3ccccc3)=O)C(CC3CC3)C2)=O)cc([N+](=O)[O-])n[nH]1 12967,c1(NC(=O)NC2C(C)(C)C2)cccc(CN2CCOCC2)c1 12968,C(C)(CCC(=O)NC1CN(C(c2cncc(N)c2)=O)CC1c1ccccc1)OC 12969,c1(C(N2CCN(C(c3c(CC)onc3)=O)C(CC#N)C2)=O)ccc2ccoc2c1 12970,C1(NC(C(=O)OC)c2csnn2)CCCC1(C)C 12971,C1(NC(=O)NCC(C2CCOCC2)(C)C)CC2(C1)CC(F)(F)C2 12972,c1(C(=O)NC(C=CC(=O)NC2(C)CC(=C)C2)C)cc(C)ccc1O 12973,C1(C(=O)NC2(C)CC(C(=O)OC)C2)CNC(=O)CN1C(=O)CCc1ccco1 12974,Cc1cc(NCC2(O)CCCN(C(C3(O)CC3)=O)C2)n2ncc(C)c2n1 12975,C#Cc1c[nH]nc1C(=O)NCC=CCNC(C1CCC(NC(C)=O)CC1)=O 12976,C(CCC#N)(C(=O)O)NC(CNC(c1ccc(C)o1)=O)=O 12977,C1(C(N(C)CC2CCCN(C(c3cc(CO)on3)=O)C2)=O)CC2(CCCC2)CO1 12978,C1(NC(=O)OC(C)(C)C)CC(C(=O)NCCc2ccno2)C12CCC2 12979,c1(CNC(C(C)O)=O)cn(CC2CCCN2C(c2cc(C(F)F)on2)=O)nn1 12980,N1(C(C(CCCC)C)=O)CCCC2CN(C(=O)COC)CC12 12981,c1(N2CC=CC(NC(C3C(CC)CCC3)=O)C2)ncnc2sc(C)nc12 12982,C=CC1(C(=O)NC(c2ccc(O)cc2)C)CCN(C(C2CC=CCC2)=O)C1 12983,c1(C(=O)NCC(CNC(CCn2ncc(C)c2)=O)C)cn(C)nc1C 12984,CCCCC(F)(F)C(=O)NCCCC1CN(C(C2Cc3nccn3C2)=O)CCO1 12985,c1(C(=O)NC2CC(C)(C)N(C(C3COC(=O)O3)=O)C2)cccc([N+](=O)[O-])c1 12986,c1(NC(C(C2CCN(C(c3sccc3Cl)=O)C2)C)=O)ccc2c(c1)OCC2 12987,N1(C(C(CCCNC(C2CCC3CC23)=O)O)=O)CC=CC12CCCCC2 12988,N1(C(C2CC3(C2)C(=O)N3)=O)CCN(C(CC=C)=O)CC(C)(F)C1.C(C)(C)(C)SC 12989,N1(C(C=C(C)C(C)C)=O)CC2CCCC2(NC(=O)CNS(=O)(=O)c2cccs2)C1 12990,C(C(CC(C)C)NC(=O)C(C)O)NC(CCCN(CCC)CCC)=O 12991,N1(C(C=COCC)=O)CC(C)CN(C(C2CCSC(C)C2)=O)CC1C 12992,C(=O)(C1CC(NC(=O)C(N2CCOCC3(CC3)C2)=O)c2ccccc21)OC 12993,c1(C(=O)NC2CCCN(C(C3(C)CC(C)C3)=O)C2)cccc2c1NCC(C)C2 12994,c1(C(=O)NCC2N(C(C(C)C3CCCC3)=O)CCCC2C)nccc2occc12 12995,c1(C(N(CCCNC(C2CCC(C(F)(F)F)CC2)=O)C)=O)ncn2c1COCC2 12996,C12(C(=O)NCc3c(Cn4cc(CNC=O)nn4)nco3)CCN(CC1)C2 12997,c1(C(N2CCCN(C3COC(C)(C)OC3)CC2)=O)cc(O)nc(Cl)c1C#N 12998,c1(C(CN2CCC(N(c3ccc(C)cc3)C)C2)=O)ccc(C)c2cccnc12 12999,N1(C(C2C(C)(C)C2)=O)CCC(COC2CCN(C(=O)CN3CC4CC4C3)C2)CC1 13000,Cc1cnc(NC(C)CC(C)C)c(S(=O)(=O)N2CC(CO)C3(CC3)C2)c1 13001,c1(SC)cc(N2CC(CN(C(=O)CC3SC(=N)NC3=O)C)C2)nc(SC)n1 13002,N(C)(C1CCCc2ccccc21)Cc1c(OC)cccc1Br 13003,C1(NC(c2cncs2)=O)(CNC(C23COC(CF)(C2)C3)=O)CC2CCC1C2 13004,C1(NC(C=C(CCC)C)=O)CCCCC1N=c1nc(C2CCCC2)[nH]s1 13005,c1(C(=O)NC(CNC(COCCCCC)=O)(C)C)cc(N)c(C)cc1Cl 13006,N1(C(C2CC(SC)C2)=O)CC(NC(c2ccc(-c3cccs3)s2)=O)CC(C)C1 13007,N1(C(c2cc(SCCCC)c(Cl)cc2)=O)CCCN(C(C2CCCC2)=O)CC1C 13008,c12cc(Cl)ccc1OC2.N1(C(C)=O)CCC(NC(=O)Cc2cc(N(C)C)no2)C1 13009,c1(C(C)(C)C)nnc2n1CC(NC(=O)C(=O)N(c1ccc(O)cc1)CCO)CC2 13010,Cc1cc(C)c(C(=O)NCC(C)(C)CNC(=O)C(C)N(C)C)c(N)c1 13011,C#Cc1ccc(NC(C2(F)CCCN(C(C3CCCN3C3CC3)=O)C2)=O)cc1 13012,c1(C(C)NC(=O)NCC2(c3cccc(Cl)c3)CCOCC2)nc(Cl)ccc1Cl 13013,N1(C(C2(OC)CCCCC2)=O)CCC(C)C(NC(c2cc(F)ccc2Cl)=O)C1 13014,C1(C(N(CCCSC)C)=O)C(NC(c2cc(C3CC3)[nH]n2)=O)C1(C)C 13015,N=c1[nH]c2ccc(C(N3CC(NC(c4cc(CO)on4)=O)CC(F)C3)=O)cc2o1 13016,N1(C(c2cnco2)=O)CC2CCC(CNC(C34CCC(CC3)CO4)=O)C2C1 13017,C(=O)(C(F)C(=O)NC1(C)CC(NC(=O)CC2CC2(C)C)C1)OCC 13018,c1(N(C(=O)COC(C)C(F)(F)F)CCOC)sc2ccccc2c1Cl 13019,CC1CCCCC1(C)C(N1CCC(c2cn(CCC3CCOC3=O)nn2)C1)=O 13020,N1(C(C(C)CNC(c2cc(C3CC3)on2)=O)=O)CCC2CCN(C)CC12 13021,N#Cc1cn[nH]c1C(N1CCC(N(C)C(C2CCCCO2)=O)CC1)=O 13022,C1(NC(C(CCC)NC(C)=O)=O)CN(Cc2ccncc2Cl)CC(F)(F)C1 13023,c1(SCC)cnc(O)c(C(N2CC(CNC(=O)CC(C)C)CC2C)=O)c1 13024,Cc1ccc2nc(N3CCCC(C(C)NC(c4cn(CCO)nn4)=O)C3)sc2n1 13025,c1(C(N(C2CC(NC(C(C(C)(C)C)OC)=O)C2)C)=O)cc(C)c(=O)n(C)c1 13026,N1(C(c2c(SC)scc2)=O)CC2(C)CN(C(=O)C=CCO)CC2(C)C1 13027,Cc1csc(=O)n1CC(N1CCN(CC(C)(C)F)CC1)=O 13028,C1(C)(CO)CCOC1.C(C)(C(=O)NC1CN(C(COCOC)=O)C1)O 13029,C1(NC(CNC(=O)OC)=O)COC2(CCN(C(=O)CSc3ccoc3)C2)C1 13030,c1(OC)c(NC(N2CCCC(C)C2C(=O)O)=O)ccc(F)c1Br 13031,Cc1ncc(C=CC(=O)NCCCCCN(C(=O)CN(C)C2CC2)C)c(O)n1 13032,C(c1cccnc1)=CC(=O)NCc1ccc(C(=O)NC2CC(O)C2)nc1 13033,c1(C(=O)NC2CC(C)(NC(C3C(C)OC(=O)N3)=O)C2)cc(N(C)C)ccc1F 13034,CCC(O)C(F)(F)C(=O)N1CCCC(CCC(=O)NC2C(O)CC2O)C1 13035,CCCCC(O)C(C)C(=O)NCC(C(N1CCOC(C)CC1)=O)N(C)C 13036,C1(COCC(=O)NCC(C)(C)NC(C23CCC2C3)=O)CCCCO1 13037,c1(OC)cc(CC(N2CC(CNC(c3cnc(C#N)s3)=O)CC2C)=O)ccn1 13038,c1(C(N2CCC(NC(CNS(N)(=O)=O)=O)CC2)=O)cc(Cl)ccc1Cl 13039,c1(OC)ccc(Br)c(CN=C(NCc2ccco2)NCC2(F)CCOC2)c1 13040,Cc1nc(-c2ccccc2)ncc1C(=O)NC1CN(C(C2CCCC(O)C2)=O)C1 13041,c1(C(=O)NCCCN(C(=O)CC2CC2(C)C)Cc2ccccc2)snc(O)c1Cl 13042,C(C(=O)N1CC2C(C(=O)NC(C)(CO)C3CCC3)C2C1)(C(C)(C)C)OC 13043,Cc1cnc(C(C)NC(=O)C=CC(C)(C)NC(=O)CCCNC(=O)OC)s1 13044,c1(CC)n[nH]c(=NC2CC3CN(C(=O)Cc4cc(C(F)(F)F)co4)CC23)o1 13045,N(C1CCOc2ccc(F)cc21)Cc1ccc(-c2ccc(N)c([N+](=O)[O-])c2)s1 13046,C(=O)(CC(C)CC(C)C)N1CCC(C(N(CCN(CC)CC)C)=O)(CO)C1 13047,C1(NC(c2c(Cl)cn(CCC)n2)=O)CCC12CN(C(=O)C(C1CCCCC1)O)C2 13048,CS(=O)(=O)c1cnc(O)c(C(=O)NC2CCN(C(c3ccnnc3)=O)CC2O)c1 13049,N1(C(CC2CC(=C)C2)=O)CCN(CC(C)NC(=O)CC2(Nc3cn[nH]c3)CC2)CC1 13050,N1(C(CSCC(C)C)=O)CCC2(C1)CN(C(=O)C(N1CCC(C)C1)=O)CCO2 13051,N1(C(c2cc(CCOC)on2)=O)CCC2(CCCN2C(=O)CP(C)(C)=O)C1 13052,N(C1CCc2cccnc21)C(N(C)Cc1ncc(Br)cc1Cl)=O 13053,c1(C(=O)NC(CNC(C(n2ccc(C)n2)C)=O)CO)cnn2cc(C#N)cnc12 13054,C1(CNC(c2ccc(-c3cc[nH]n3)s2)=O)CCC(NC(C2(CF)CCC2)=O)CC1 13055,C12(CNC(C(C)NC(COC)=O)=O)CC1CN(C(C1(F)CCCCC1)=O)C2 13056,N1(C(c2cc(C(CC)C)no2)=O)CC(F)(F)CC1CCNC(=O)CCSC 13057,c1(COC)ccccc1NC(C1(COC)CCN(C(=O)C(C)n2cnnn2)C1)=O 13058,N1(C(C2CCCN(C)C2)=O)CCC(CNC(C2CC(=O)N(C)C2)=O)C12CC2 13059,C1(CN(C(CN(C)CC)=O)C)COCCN1C(=O)CCCc1csc(C)n1 13060,c1(NCCCC(C)O)ncccc1S(=O)(=O)N(CCCN(C)C)C 13061,C1(NC(c2cnc(C)[nH]2)=O)COCCN(C(c2cn(CC3CC3)nn2)=O)C1 13062,N1(C(C=CC(C)NC(C2CCCS2)=O)=O)CC2(CCNC(=O)O2)C1 13063,c1(OCC)ncc(NC(C2CCCC(NC(c3cncc(C)c3)=O)C2)=O)cn1 13064,C(CNC(=O)CCOC1CCC1)(C(=O)N(C)CCn1cccn1)OC 13065,C#Cc1ccc(C(=O)NCCOCCC(N2CC3CC(CO)C(C3)C2)=O)c(C)c1 13066,c1(NC(c2nn(CC)cc2C)c2n(CCC)nnn2)ccc(C(=O)OC)c(Cl)c1 13067,c1(C(CNC(C2CNC(=O)C2)=O)NC(=O)NC(CC=C)C)ccccc1OC 13068,C(=O)(C(C)(C)CC(F)F)N1CC2C(NC(Cc3c(C)n[nH]c3)=O)(CC2)C1 13069,C(=O)(C1COc2ccc(F)cc21)N1C(CCNC(CCOC)=O)CCC1 13070,CCCCC(CC)C(=O)NC12COC(C1)C(NC(C1(COCC)CC1)=O)C2 13071,c1(C(=O)NC2CCC(NC(C3(C)CCC(=O)N3)=O)C2)cccc2c(C#N)c[nH]c12 13072,c1(OC)nnc(Cl)cc1NC(=O)Cc1ccccc1NC(c1sccc1C)=O 13073,CCC(C)CCC(O)CC(=O)NCCC1CCN(C(=O)CS(=O)(=O)C2CCCC2)C1 13074,C=C(C)C(C)(C)C(=O)NC1CC1NC(C1CCN(Cc2cccnc2)CC1)=O 13075,C1(NC(CCC=C)=O)CC12CCN(C(=O)Cc1cnccc1C(F)(F)F)CC2 13076,N1(C(=O)CSc2cccs2)CCCC2CN(c3nc4ccccc4o3)CCC12 13077,c1(C(=O)NC2CN(C(C(CCOC)OC)=O)CC2O)cc2cc(C)ccc2[nH]1 13078,C(C)(CCC(=O)N1CC(C(F)Cn2cc(CC3CCCC3)nn2)C1)OCC 13079,c1(NC(c2ccc(NC(C)=O)cc2)=O)n[nH]c2c1CN(Cc1cc(Br)c(C)s1)C2 13080,N1(C(c2cnc(C)[nH]2)=O)CCC(C2CCCN(C(c3nc(C)c(C)s3)=O)C2)C1 13081,N1(C(Cc2cc(OC)c(F)cc2)=O)CCN(Cc2ccc([N+](=O)[O-])o2)CC12CC2 13082,C(=O)(C(C(C)O)N(C)C)NCC(CNC(=O)CCc1ccsc1)OC 13083,C1(O)(CCC)CCN(C(=O)C(C)(C)CNC(=O)C(C)OCCOC)CC1 13084,c1(CCCOC)cccc(Br)c1.C12(CNC(=NC)NCC)CCN(CC1)C2 13085,N1(C(CCOCCC)=O)CCC(O)(Cn2cc(CN(CCOC)CC)nn2)C1 13086,Cc1cc(=NCc2nnc(C(C)(C)C)s2)[nH]c(N2CC(=O)NC(=O)C2)n1 13087,C=C(F)C1(CC(=O)NC(C)(C)C(C)NC(C2CC2(C(C)C)CC)=O)CCC1 13088,C1(N(C(CC)=O)C)CCCCN(C(C23CC(c4ccc(OC)cc4)(C2)C3)=O)C1 13089,c1(CN2CCC(C(C(=O)NC(n3ccnc3)C)C)CC2)ccc2c(c1)CCO2 13090,c1(OC)ccc(C(N2CC3CC(NC(C4CCC(=O)CC4C)=O)C3C2)=O)c(C)c1 13091,c1(C(C)=O)ccc(OC(C)C(N2CC(NC(C3(CO)CC3)=O)C(O)C2)=O)cc1 13092,c1(C(C(=O)NCC(CNC(=O)C=CBr)F)OCC(F)(F)F)ccccc1 13093,C1(CC(N2CCC(N(C(=O)C=CCOC(C)(C)C)CC)C2)=O)CC(C2CC2)C1 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13214,N1(C(CN(C)C(N)=O)=O)CC2(C1)C(NC(C1CCC3CCC1O3)=O)CCS2(=O)=O 13215,Cc1cc(C(N2CCC2CNC(c2cc(-c3ccco3)no2)=O)=O)cn1C 13216,c1(C(C)=O)c(CC(=O)NCC(C)(C)NC(=O)Cc2cscn2)c[nH]c1C 13217,c1(C(=O)NC2(CNC(C(CC(C)C)F)=O)CCC2)cc(F)c(C(F)(F)F)cc1F 13218,c1(C(C(=O)NCCCCCC)N(C2COC(=O)O2)C)ccc([N+](=O)[O-])cc1OC 13219,C1(CC)CN(C(=O)CN2CCNC(=O)C2)CCN1C(=O)CC1CCCCC1O 13220,c1(C(N(C2CCN(C(C3CCCS3)=O)CC2)CC)=O)n[nH]c2c(C)cccc12 13221,c1(C(=O)NCC(C(C(C)C)C)NC(c2nsnc2O)=O)cc(F)c(F)c(F)c1F 13222,c1(CC(=O)NC2CCC(CNC(C(C)(F)F)=O)C2)cccc2cnccc12 13223,C(=O)(C1=NOC2(CCC2)C1)NC(C)(C)CCCNC(C1(C)CCC(=O)NC1)=O 13224,C1(C(N2CC(NC(=O)NC)C2)=O)C2CC(O)C1N(C(c1ccnn1C)=O)C2 13225,C(=O)(C(CC)(CC)CC)N1C2C(NC(C3N(CC)CC3)=O)CC(C2)C1 13226,C=CCC(C)(CNC(=O)CC1CCCCN1C(c1nnn(CC)c1C)=O)CO 13227,c1(C(=O)NC(C2CC(C(=O)Nc3ccsn3)C2)C)c[nH]nc1-n1cnnn1 13228,C1(NC(c2cn(CCNC(C3(CC)CC3)=O)nn2)=O)CCCCC1O 13229,C1(NC(C2C=CCC2)=O)C=CCN(C(=O)CC(c2ccccc2)c2ncc[nH]2)C1 13230,CC1(C)CCC(O)(CNC(=O)CCN(C(=O)CCCC2CC2)CCCO)C1 13231,c1(CN2CCC(N3CCN(c4cc(CC)ncn4)CC3)C2)cccn2nccc12 13232,CC1CN(C(c2ncn3c2CCCC3)=O)CC(C)C1NC(c1ccc[nH]1)=O 13233,CS(=O)(=O)CC(=O)NCC1(C(=O)Nc2ccc(F)nc2)CC12CCC2 13234,C1(F)(C(=O)NCCC(C)F)CN(C(C2CCC2C#N)=O)C1 13235,c1(C(N(C2CCN(C(c3ccsn3)=O)C2)C)=O)cccc(C=O)c1Br 13236,C(CC(=O)C(C1CCNC1(C)C)=O)(C(F)(F)F)N1CC(C)(C)C1 13237,N1(C(C(C2(O)CCC2)NC(c2ccc(NC)cc2)=O)=O)CC2(CCC(O)CC2)C1 13238,c1(COC)noc(C(=O)N(C2CCC(NC(C3CCC3)=O)C2)C)n1 13239,c1(NC)ccnc(C(N2CCC(CNC(=O)CCC(C)c3ccccc3)C2)=O)c1 13240,C(=O)(CCCC(=O)NCCCC(C)(C)NC(C1CC2CCC1C2)=O)NCC 13241,N1(C(c2cc(C)nnc2O)=O)CCC(N=c2cc(C)nc(S(C)(=O)=O)[nH]2)C(C)C1 13242,N1(CC(=O)NC(C)CCNC(=O)Cn2nnc(C3CC3)n2)CCC(N(C)C)CC1 13243,c1(C(=O)NCC(N2CCC(OCCC3CC3)C2)=O)c(C(=O)CCl)cccc1F 13244,c1(C(N(C2CN(C(c3ncncc3Cl)=O)C2)C)=O)ccnc(C2CC2)c1 13245,Cc1cccc(CN(CC(C)C#N)Cc2ccc(OCF)cc2)c1C 13246,N1(C(C2CCC(C)(CC)O2)=O)CC=C(CC(=O)NCc2ccc(F)c(O)c2)CC1 13247,N1(CC2C(C(=O)OCC)CCN2)CCCC(C)(O)C1 13248,C1(CNC(c2nn(CC)nc2C)=O)(NC(C2CC(O)C2)=O)CCCCC1C 13249,c1(C(=O)NC2COCCN(C(C(CCSC)O)=O)C2)cc2ncccc2s1 13250,c1(C(=O)NC(C2CCN(C(C=CCC)=O)C2)C)c(C)cnn1C 13251,c1(CC(N2C(CCNC(=O)Cc3ccno3)CCC2)=O)ccc2ncsc2c1 13252,C(CC(C)C)(C(=O)NC1(CNC(C2CCOC2)=O)CC1)OC 13253,C1(C(=O)NCC(CNC(=O)C2CC2)OC)CC2CCC(C1)N2S(C)(=O)=O 13254,C(C(C)C(=O)N(C1CCC1)C)N(C(CCNC(C)=O)=O)C 13255,C1(NC(C(CC=CCC)C)=O)C2CCC(C2)C1C(=O)NCC1CCC(C)C1 13256,c1(C(=O)NC(c2cccnc2N(C)C)=O)ccc(C2CC2)c(Br)c1.C12CN(C1)C2 13257,C1(C(=O)NCC(C)(C)C(F)F)CN(C(=O)CC2CC(C3CC3)C2)C2(CCC2)C1 13258,N1(C(c2c(CC(C)C)n(C)nc2)=O)CC(NC(C2CNC(=O)C2)=O)CC(C)(C)C1 13259,C(=O)(C1CCc2c[nH]nc21)N1CCCN(C(C(CCC)(C)O)=O)CC1 13260,c1(C(=O)NCCCN(C(c2cnc[nH]c2=N)=O)CC)ccc(F)cc1OC 13261,C1(C(C)OC)CCN(C(=O)C=CC(C)NC(=O)C(C)C2CCCC2)CC1 13262,N1(C(c2c(CC)noc2)=O)C2CCC1C(NC(=O)CCc1ccc(Br)cc1)C2 13263,C1(CCC)CN(C(=O)C(C)(C)n2cccn2)CC1NC(C1C=CCC1)=O 13264,N1(C(c2c(CC)nns2)=O)CC(C(=O)NC(C)(C)CCCO)C(F)(F)C1 13265,N1(C(CCN(C(C2=CCCC2C)=O)CCO)=O)CCCN2CCCC2C1 13266,Cc1cccn2c(CC(=O)NCC(CC(C)C)NC(=O)CCC(C)(C)C)cnc12 13267,CN1CCN(C(c2cc(O)n(C)n2)=O)C(C(N2CCCC(OC3CC3)C2)=O)C1 13268,c1(CN2C(C(=O)NCc3ncc(Br)s3)CC(O)C2)c(Cl)ccnc1Cl 13269,C1(=O)CC(C)(C)C(CC)CNC2C(CNCc3ccc(C(=O)NC)o3)CCN12 13270,N1(C(c2cc(C(C)=O)[nH]n2)=O)C(CNC(=O)C(C)(C)C2CCC2)CC2COCC12 13271,c1(-c2ccc(Sc3ccc(CC)cc3)cc2)n[nH]c(=NC(=O)Nn2cncn2)s1 13272,C(N=c1[nH]c(=NCc2[nH]nnc2C)c2ccccc2[nH]1)c1ncc(C)o1 13273,C(CCCC(=O)O)n1cc(SCCNC(C(c2ccnn2C)C)=O)nn1 13274,Cc1c(CC(N2CCOC(C(=O)NC3CCCC3F)C2)=O)cnn1C 13275,C(CS(=O)(=O)C1CCOCC1)NC(CCC)C1CCC1 13276,C12(CN(CCOC)C(C3CC3C(=O)NC(C)=O)=O)CCC(C1)C2c1ccccc1 13277,CC(C)CC(O)CC(=O)N1CCC(C(C)(C)CNC(C2CCOC2)=O)CC1 13278,C#Cc1c[nH]nc1C(=O)NC1CC1NC(c1ccccc1COC(C)(C)C)=O 13279,N1(C(CCCC)=O)CCC(NC(c2csc(-c3ccco3)n2)=O)C(CC)C1 13280,c1(C(=O)NC2CC3(CN(C(C(C)CN(C)C)=O)C3)C2)nnc(O)c2ccccc12 13281,N1(C(C2CC=CC(NC(C3(CO)CCCCO3)=O)C2)=O)CC2C=CCC(C2)C1 13282,c1(C(=O)NN2C(C3CCCCC3)CCC2)cn2ccnc2cn1.c1(C)ccccc1 13283,C1(C(N(C(C)C(=O)NC2CCOC2)CCC)=O)CCCC(C#N)C1 13284,Nc1ccc(C(N2CC(NC(=O)C(F)C(F)(F)F)C2)=O)nc1C(F)(F)F 13285,C(C(CC(C)C)NC(=O)C=C(C)c1ccco1)NC(c1n(CC#C)cnn1)=O 13286,C1(NC(CCC2(C)CN(C(c3c(CCC)[nH]cc3)=O)C2)=O)(CO)CCCCC1C 13287,C1(C(N(C2(CC=C)CCOC2)C)=O)CN(C(=O)CC2CCCC3CC23)CC1CC 13288,CC1CC(=O)NCC1C(N1CCC(C)(CNC(=O)CC2(O)CC2)CC1)=O 13289,C1(O)(C(=O)NCCCn2cc(C3CCCO3)nn2)Cc2ccccc2C1 13290,c1(CC2(NC(c3cncc(OCC)c3)=O)COC2)ncnc2cc(Br)ccc12 13291,C(=O)(C1CCCc2sccc21)NCC1(NC(C2CCN(C)C2)=O)CC1 13292,Cc1cccc(CN(C(=O)C(CCC2CC2)NC(=O)C(C)c2cc[nH]n2)C)n1 13293,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC1CC1CNC(C1CCC2(CCC2)C1)=O 13294,c1(OC)cc2nn[nH]c2cc1C(=O)NCCCCNC(c1cnn(C)n1)=O 13295,C1(CCC(=O)NCCCN(C(c2nccn2C(C)C)=O)CC)CCN(C)CC1 13296,c1(C(N(C)CC2(CNC(C3C(CC)C3)=O)CC2)=O)ccnn1CC 13297,c1(CC(=O)NCC2C(NC(C3(C)CC3)=O)CCC2)ccc2nonc2c1 13298,C1(C(=O)NC(C23CCC(CC2)C3)C)(NC(C2CCO2)=O)CCCCC1 13299,c1(C(N2CC3CC3(C(=O)NCc3cncs3)C2)=O)cc(Cl)c(O)cc1F 13300,C#CC12CCN(CC1)CC(=O)N2.C(C(C)(C)C1CC1)N(C)C 13301,CC(C)C(F)(CNC(C1(CCN(C)C)CC1)=O)C(=O)NCC(C)(C)CN=[N+]=[N-] 13302,n1(CCC(N2C(C)CN(C(C3(CO)CCOC3)=O)CC2)=O)ccc2ccccc12 13303,C1(C(N2CC(C)(NC(CC(=O)NCC#C)=O)C2)=O)CC(C2CCCC2)C1 13304,C(CC1=CCN(C(c2ccc(F)c(F)c2N)=O)CC1)NC(C=CC(CC)=CC)=O 13305,c1(N(C)C)ncnc(N2CCC(OCCNC(c3ccco3)=O)C2)c1[N+](=O)[O-] 13306,c1(C(=O)OCC)nnn(C)c1CNCc1cscc1Cl 13307,C1(C(=O)NC(CC=C)C(=O)OCC)CNC(=O)CN1C(C1CC1C(F)F)=O 13308,n1(CC)ccc(CNC(=O)CC2(OC)CN(C(=O)CC(O)c3ccccc3)C2)n1 13309,C1(CC(N2CCN(c3nc(C)cc(C)n3)C(C)C2)=O)CCCC2CCCCC12 13310,Cc1ncccc1C(N1CC(C(N)=O)(CNC(=O)CC2CCCC(C)O2)C1)=O 13311,c1(C(=O)NCC(CC)NC(C2NC(=O)CC2C)=O)ccc(N)cc1O 13312,C1(C(=O)NCCOCCC(=O)NC(CC)C2CC2)CCC1C#N 13313,c1(OCCOC)cc(F)c(F)cc1-c1c[nH]nc1-c1c(OC)nc(Cl)c(Cl)n1 13314,N1(C(C2C(CNC(C(N)=O)=O)CCO2)=O)CC2(CCC2)CC1CO 13315,C1(CC#C)(C(=O)NC(CC(N)=O)C2CC2)CCN(C(c2ccnn2C)=O)C1 13316,c1(OC)cc(C)nc(NC2CC(NC(=O)COCc3nnc(C)s3)C23CCC3)n1 13317,O=C1NCCCCC1S(=O)(=O)N1CC2CCCC(C1)N2c1nccc(CO)n1 13318,N1(C(c2ccc(OC)nn2)C(=O)NCCOC)CCS(=O)(=O)C2(CCC2)C1 13319,N1(C(C(CC#C)C)=O)CCOC2CN(C(=O)Cc3cccc(OC)c3Cl)CC12 13320,C1(NC(C2CC(O)(c3ccncc3)C2)=O)CCC(NC(C2CCOCC2)=O)C1 13321,Cc1ncc([N+](=O)[O-])cc1NC(=O)CC1CCN(Cc2cc(F)c(F)c(F)c2)C1 13322,O=CN1CCCN(C(=O)CC(CC2CC2)NC(=O)COC2CCOC2)CC1 13323,c1(C(=O)NCC(C)N(C(CN(CC)CC)=O)C)coc2cccc(Br)c12 13324,C(CC)(CCCO)N(C(=O)C(C#N)CC)C(=O)CC1(C2CC2C(F)(F)F)CCC1.CC 13325,c1(OC)ccc2[nH]ccc2c1C(N1CCC(C)(NC(=O)C(CC(C)C)OC)C1)=O 13326,C(=O)(C(C)(C(C)C)OC)NC(CC=C)CNC(c1n[nH]c(C)n1)=O 13327,c1(C(=O)NC2C(C)CN(C(=O)CCC3(C)CC3)C2)ccc(N)cc1Cl 13328,C=CCC(CC)C(=O)N1CCN(C(C2(C(=O)OC(C)(C)C)CC2)=O)CC1COC 13329,Cc1ccc(O)cc1C(N1CC(C)CC1C(=O)N(C1CC2CC2C1)C)=O 13330,c1(CC)nn(C)cc1C(=O)NC1CC(CNC(=O)C(C)(C)NS(C)(=O)=O)C1(C)C 13331,CC1(C)C(NCC(F)(F)C(F)(F)F)C2CCCN(C(C3CC34CCCC4)=O)C12 13332,Cc1ccc2sc(C(N3CCN(C(=O)C(C4CC4)N(C)C)CC3)=O)cc2c1 13333,CC1CCN(C(C2CCCCO2)=O)CCN1C(c1ccn2ccccc12)=O 13334,C(CN=c1[nH]c(=NC2CCC(C(N)=O)CC2)c2ncccc2[nH]1)NS(NC)(=O)=O 13335,CC(CO)(C(=O)NC(C1CCCCC1)CO)NC(=O)CCC1CCOCC1 13336,N1(CCc2cn(CCC=C)nn2)CCOC(Cc2ccccc2)C1 13337,c1(COC)cnc(NC(=O)NCC(c2ccccn2)C)nc1 13338,CC1CN(C(=O)C(=O)C(F)(F)F)CCC1NC(=O)CCC1CC1(Cl)Cl 13339,C1(CC(=O)N(CC(C)NC(=O)CCCCCn2cnnn2)C)CCS(=O)(=O)CC1 13340,CCC(CC)C(=O)NC1CC(CO)N(C(=O)CNS(C)(=O)=O)C1 13341,CC1CC2CN(C(C3CC3(Cl)Cl)=O)CC2N1C(=O)C(O)CC(N)=O 13342,C1(OCC(N2CC(Oc3ccsc3)C2)=O)CCN(C(C23C=CC(CC2)C3)=O)CC1 13343,C1(C(=O)NC(c2ccnc(F)c2)C)CCCCCN1C(c1ccc(C(N)=O)o1)=O 13344,CCC(C(=O)N(CC(C)O)CCNC(=O)CC1CCCO1)NC(c1ccco1)=O 13345,C1(C(N2CCCC2CNC(C23CC(F)(C2)C3)=O)=O)CCN(CCO)C(=O)C1 13346,C1(NC(C(C)OCC)=O)CN(C(c2c(Cl)csc2Cl)=O)CC1(C)C 13347,N1(C(c2cnn[nH]2)=O)CCC(NS(=O)(=O)CC2CCOC2)CC1 13348,CCCCCC(C)CC(=O)N1CCC(C)(CC(N2CC3(CO)CCC2CC3)=O)C1 13349,C1(C(=O)NC2CCC(CNC(=O)CSC3CC3)C2)CC2(CCOC2)C1 13350,C(=O)(CC(C)CNC(=O)CC(O)CN(C)C)N(CC(CC)(F)F)C 13351,CN(C)S(=O)(=O)N(C)CC(=O)NCCC1CCC(NC(=O)CC2CC(F)C2)C1 13352,c1(OC)cc(C(F)(F)F)c(OC)cn1.N12CCCC(C1)Oc1csc(n1)C2=O 13353,c1(C(=O)NCC2(F)CC(NC(C3C(OC)CCC3)=O)C2)oc(CO)nc1C 13354,C1(NC(c2ccnc(C)n2)=O)C2CC1CN(C(=O)CSc1ccccn1)C2 13355,CC1CCC(CNC(=O)C(O)C(F)(F)F)CN1C(c1cnc[nH]1)=O 13356,CC(C#N)CCC(=O)N1CC(CNC(c2cc(-c3cnn(C)c3)on2)=O)C(O)C1 13357,C1(C)(CNC(=O)NC(CC)C(=O)N2CC(COC)(OC(C)(C)C)C2)C=CCCC1 13358,C1(NC(C2CC(=O)N(C3CC3)C2)=O)CCN(C(C2C(C(=O)NCC#C)C2)=O)CC1 13359,c1(C(=O)OC)cnc(N2CCC(OCCNC(C3CC=CCO3)=O)C2)s1 13360,C1(C(=O)NCC(C(C)C)O)CN(C(C2CS(=O)C2)=O)CC1(C)C 13361,c1(CC)c(C(=O)NCC2CCCN(C(=O)C(C)Cn3cccn3)C2)cnn1C 13362,C(=O)(C(CO)C(C)C)NCC(C)N(C(Cc1cccc(C(C)C)c1)=O)C 13363,c1(OC)ccc(C(=O)NCCNC(=O)CC2CCCC(C)C2)nc1Br 13364,N1(C(CC(CC)C(C)C)=O)CCCC2(CCN(C(=O)C(C)(C)C(O)CF)CC2)C1 13365,C1(NC(c2c(C)cns2)=O)CCC(CNC(c2csc(Br)n2)=O)CC1 13366,C1(C(=O)N=c2ccnc(Br)[nH]2)CC(c2cccnc2)=NO1 13367,CC(C)C(CNC(=O)C=C(C1CC1)C1CC1)C(=O)N1CCC(O)(C(N)=O)C1 13368,Cc1c(CC(=O)NCCCCN(C)C(c2ccnn2C)=O)ncn1C 13369,N1(C(C(C)NC(C)(C)C)=O)CC2(C1)SCCC2NC(=O)CCCC(N)=O 13370,CC1CN(C(c2cccc(F)c2)=O)CCC1C(=O)NCc1ccc(O)nc1 13371,C1(C(N(CC(CCC)O)C)=O)(CNC(c2c(C)cnn2C)=O)CC12CCC2 13372,C1(C(N2CCN(c3cncc4nccn34)CC2)=O)CC2(C1)CC21CCC1 13373,c1(OC)cc(NC2CCN(CC(=O)O)CC(F)(F)C2)c([N+](=O)[O-])c(F)c1 13374,N1(C(C2CCCN(C(N(C)C)=O)C2)=O)CCC(NC(=O)C(F)=C(C)C)C12CC2 13375,N1(C(C(CC)NC(N)=O)=O)CC2CCC1C(NC(=O)C(c1cccnc1)NC)C2 13376,C12(CNC(C(CC)N(C)C)=O)CC1CN(C(C1COCCO1)=O)C2 13377,C1(CC(N2CCC(NC(CCC#C)=O)CC2C)=O)CSc2ccccc2O1 13378,c1(NC(c2cnc(-c3cccs3)s2)=O)ccc(F)c(-c2nc[nH]n2)c1 13379,C1(C)CCC(=O)OCCO1.c1(CNC(C)=O)cccc(CNC(=O)NC(C)C)c1 13380,c1(CC(=O)NCCCC(C)NC(c2ccoc2)=O)cccc(OC(F)(F)F)c1 13381,N1(CC(=O)NC2CCC2NC(C2(CC(F)F)CC2)=O)Cc2ccccc2C1 13382,Cc1nc(O)nc(O)c1CC(=O)NC12CCCC1N(C(=O)C(=O)C(F)(F)F)CC2 13383,N1(C(CC(CC)(C)C)=O)CCCN(C(c2ccc(OC3CCC3)cc2)=O)CC1C 13384,CC1CCC(CNC(=O)C(Cn2cccn2)NC(=O)CC23CCC(CC2)C3)N1C 13385,C1(C(c2ccccc2)C(=O)NCCN(CCC(C)C)CCOC)CCCCCC1 13386,c1(C(=O)NCC(CC)NC(c2ccn(-c3cccc(F)c3)n2)=O)cccnc1C 13387,C12(C(=O)NCCCN(C(=O)CN3CCCS3(=O)=O)CC)CCCCC1C2(F)F 13388,c1(COC)nc(NCCCS(C)=O)cc(=NCC2(CS(C)(=O)=O)CCC2)[nH]1 13389,N1(C(COCCCC)=O)CCC(C(C)(C)CNC(=O)CC2NC(=O)NC2=O)CC1 13390,CC1CC(NC(=O)CC2CCC3(CC2)CC3)CCN1CCN1CCCCCC1=O 13391,CC(C)CC(C)(CNC(=O)Cc1c[nH]nc1O)NC(C1CC(=O)NC(=O)N1)=O 13392,C1(C(=O)NCCN(C(=O)CCc2cnoc2)CC)CCC(=O)N1CCC(F)(F)F 13393,C1(OCC(=O)NC2CC(NC(Cn3ncc(C(=O)OC)c3)=O)C2)CCCCC1C 13394,C1(NC(C2=C(C)CC2)=O)CN(C(c2csc(CO)n2)=O)C2CCCC12 13395,CCC(CC(=O)NCC1(O)CCN(C(=O)COC2(C)CCCC2)C1)CC(F)(F)F 13396,C(=O)(CC(C(=O)N(C(C)CNC(=O)CCCC(C)=O)C)NC(=O)OC)OC 13397,N1(C(C(C)NC(=O)OC)=O)CCC(NC(C2CCC2)=O)C(CO)CC1 13398,Cc1cc(C)c(C(=O)NCCC2CN(C(C3CNC(=O)N3C)=O)CCO2)c(C)n1 13399,CCN=c1[nH]c(C)c(C(=O)NC(C2(CNC(=O)Cn3nc(C)oc3=O)CC2)C)s1 13400,c1(C(N2CC(CNC(COCCOCC)=O)C(O)C2)=O)ccc(C#N)n1C 13401,c1(C(N2CCC(NC(CC(CC)C)=O)C(F)C2)=O)cc2nc(C)ccc2o1 13402,c1(C(=O)NCC2CC(NC(C3CC34CC4)=O)CCO2)cc2ccc(F)cc2o1 13403,c1(C(=O)NCCCCCNC(COCCCCC)=O)ccc(Br)cc1O 13404,C1(CC)CN(C(C2CN(C)CCN2C)=O)CCC1NC(c1cnc(C(C)=O)s1)=O 13405,N1(C(CNC(CC(C)CN(C)C)=O)=O)CC(=O)NC(=O)C1C 13406,c12ccc(cc1)CO2.C12CCC(CC1)CN2C=O.C#CCOC 13407,CC1(C)OC(=O)NC1C(=O)NC1COCCC1NC(C1CC(F)(CF)C1)=O 13408,c1(CC)ccccc1C(=O)N(C1CCCC(N(C)C(c2ccco2)=O)C1)C 13409,c1(-c2c(C(=O)NCCCOCC)scn2)ccn(C)c(=O)c1 13410,N1(C(CC2N(C(c3cccc(NC)n3)=O)CCCC2)=O)CCC2(CC=CCO2)C1 13411,C1(F)(C(N(C)CC2COCCN2C(=O)C=CC(F)(F)F)=O)C(C)(C)C1(C)C 13412,C(C(CC(C)C)NC(C1CC(=O)N(C)C1)=O)NC(C=CC=CC)=O 13413,c1(CC)onc(C(=O)NCC2C=CCN2C(=O)C(O)C(C)C)c1C 13414,c1(CCC)c2nnn1CC1(COC)N(CC=C1)C2=O.C(=O)(CC(C)CF)NC 13415,C1(C(=O)NCC(C)CCO)CCCCS1(=O)=O 13416,c1(CNC(=O)COCCCCCC)cccc(-n2cc(-c3ccncc3)nn2)c1 13417,N1(C(C(C)(C)O)=O)CC(NC(C2CN3CCN2CC3)=O)CC(F)(F)C1 13418,N1(CCC)CCCC(C(=O)NC(C)(C)CNC(c2c[nH]c(=N)o2)=O)C1 13419,N1(C(C(C)NC=O)=O)CC(CNC(=O)Cc2ccc(F)nc2)CC1(C)C 13420,C1(Br)(C(=O)NCC(C)N(C(c2cc(CC)on2)=O)C)CC12CCC2 13421,c1(C(=O)OC(C)(C)C)cn(C)nc1CN(C(C(C)C)=O)CCCN(C)C 13422,Cc1ncn(CCNC(c2conc2C(C)NC(=O)CCn2cccc2)=O)c1C 13423,C1(CC(=O)NC2CC(NC(C(SC)SC)=O)C2)CCCC2(CC2)C1 13424,c1(N2CC(CNC(=O)C(F)CC3CCCC3)OCCC2)nc2ccc(F)cc2o1 13425,c1(CC(=O)N(CCC(C)NC(COCC(=C)C)=O)C)ccc(S(=O)C2CC2)cc1 13426,C#CCC(C)(C)C(=O)N1CCOC(CCNC(=O)Cn2ccc(C)c2)C1 13427,CC(O)C(C(=O)NCC1CCCCN1C(c1coc(C(F)F)c1)=O)N(C)C 13428,c1(C(N2CCC(C(C(C)C)NC(CCC=CC)=O)CC2)=O)cc(S(C)(=O)=O)cs1 13429,N1(C(CCCCSC)=O)C2CC1CN(C(=O)CCP(C)(C)=O)C2 13430,c1(CCC(=O)NCC(C)(C2CC2)NC(C2(F)CCCCC2)=O)nc2ccccc2[nH]1 13431,N1(C(c2cnc(CC)[nH]2)=O)CC2CC2(CNC(=O)CC2CCC(=O)N2C)C1 13432,c1(C(=O)Nc2nc(C(=O)OCC)n(C)c2)ccc(OC)nc1OC 13433,Cc1ccc2[nH]c(C(=O)Nc3ccc(CNc4n[nH]c(C5CC5)n4)cn3)cc2c1 13434,Cc1nc(NCCCOCCNC(=O)C(C(C)C)SCC(F)(F)F)cc(Cl)n1 13435,C(=O)(CCCCC(F)(F)F)NC1CC(NC(c2cc(C3CCC3)[nH]n2)=O)CC1O 13436,c1(OC)ccc2c(c1)C(C(=O)NCCCNC(c1cnc(C(N)=O)cn1)=O)CC2 13437,C(=O)(CC(C1CC1)NC(=O)C=Cc1ccco1)N(C1CCOC1)CC#C 13438,N1(Cc2nnc(CC)s2)CCCOC(CNC(c2occ3c2CCC3)=O)C1 13439,CC1CCN(C(C23CC(C)(C2)C3)=O)CCN1C(=O)C(Cc1ccccc1)N(C)C 13440,C1(NC(c2c(COC)noc2)=O)CC(CO)N(C(=O)CSCc2ccncc2)C1 13441,Cc1cc(NC(C2(C)CC(O)CN2C)=O)ccc1NC(=O)Cc1sccc1Cl 13442,C=CCCCCCC(=O)NCC(CCCC)NC(c1cc(=O)cc[nH]1)=O 13443,N1(c2n(CC=C)c(C(n3cncn3)C)nn2)CCCC(n2ccnn2)CC1 13444,C1(CNC(C(C)(F)CC2CCCC2)=O)CCCC2CN(C(=O)CC(F)(F)F)CC12 13445,C#CC1(C(=O)NCc2ccncn2)CCN(C(=O)C(=O)C2CCCC2)C1 13446,Cc1noc(C(C(C)C)NC(=O)CC2CCN(C(=O)C(C)CN(C)C)C2)n1 13447,c1(C(=O)NCC2CCN(C(CNC(C(C)(C)C)=O)=O)C2)c[nH]c(=N)nc1O 13448,C1(N(C(CCOCC#C)=O)C)CCN(C(=O)C=C(CCC)CCC)CC1C 13449,C(=O)(C(CCNC(=O)CCCCC1CC1)OC)N(C1CCN(C)C1)CC 13450,C1(=O)C(C)NCC(C)NC(=O)C=CCN1C.C(=O)(C1CC1)OC.OC 13451,C12(CCCC1)CC(=O)NC(C1CCCC1)C(=O)NC2.c1(C(=O)OC)coc(O)n1 13452,c1(C2(C(=O)NCCOCCCNC(CC(C)F)=O)CCC2)ccc([N+](=O)[O-])cc1 13453,NS(=O)(=O)CCCC(=O)NCCC1CCCCN1C(=O)CCN1CCCCC1 13454,N1(C(C(C)N(C)C(C2C3CCCCC23)=O)=O)CCC12CC(CO)C2 13455,C1(NC(CC2(CSC)CC2)=O)C2CCC(C2)C1C(=O)NCCC1CCCOC1 13456,C(=O)(C(C)C1=CCCC1)NCC1CCC(NC(c2n(C=C)ncc2)=O)CC1 13457,c1(C(=O)NCC2(F)CCN(C(CN3C(C)CCC3)=O)C2)nc2ncccn2n1 13458,c12nc3c(s1)CN(CC3)CNC(=O)N2.Cc1c(Cl)ccc(CC(O)CO)c1Cl 13459,C1(CC)CN(C(=O)CN2CCNC2=O)CC1C(=O)N(CC(C)(C)C)C 13460,C(C)(C)(CC(=O)NCCC1(NC(=O)Cc2cncnc2O)CCCC1)SC 13461,c1(C(N(C(C)CN(C(=O)CCCCc2cnc[nH]2)C)C)=O)cnc2ncccn12 13462,c1(C(=O)N(C(C2CCN(C(=O)CCSC(F)(F)F)C2)C)C2CC2)cccc(O)n1 13463,C#Cc1cccc(C(=O)NC(CNC(c2ccc(S(C)(=O)=O)o2)=O)C(C)C)c1C 13464,C#CCCCC(=O)NC1CCC(CNC(C2CCCOC2)=O)C1 13465,c1(C(N2CC(O)(CNC(c3cnn(C(F)F)c3)=O)C2)=O)ccc2cc[nH]c2c1Br 13466,c1(C(=O)NCCN(C(=O)CCC2CCCCC2)CC)nn(C)cc1SC 13467,C1(NC(c2cnc(OC)nc2)=O)CCN(C(C2CCC(N(C)C)C2)=O)CC1CO 13468,CC(C(C(=O)NC1CCOC1)N(C1CCC1C)C)C(C)(C)C 13469,C1(F)(C(N2CC(OC)C(OC)C2)=O)CCN(C(c2ccc(C(C)C)[nH]2)=O)C1 13470,c1(N2CC3CC(NCCSc4cn(C)nc4)C3C2)nc(Cl)nc2ccccc12 13471,C=CCCCC(=O)NCC(C)(C)Cn1cc(-c2ncccn2)nn1 13472,c1(C(N(C)CC2CCN(C(C3CCC(F)(F)C3)=O)C2)=O)cc2ccncc2s1 13473,c1(CC(=O)NC2CN(C(C3(CCC=C)CC3)=O)CC2C)cc(C)ccc1OCC 13474,C(N=c1[nH]c(=NCC2COCCO2)c2[nH]ccc2[nH]1)c1c(N)cccc1F 13475,C(=O)(C(F)(F)C(C)(C)O)NC1CCCC(N(C(c2c(SC)csc2)=O)C)C1 13476,C(=O)(CC(C(F)F)NC(C1(n2cnnn2)CC1)=O)N1CC(O)(CC(C)C)C1 13477,c1(CNC(C(n2cc(-c3ccccc3CN)nn2)C)=O)cccc(C(F)(F)F)c1 13478,c1(C(N(C(C)CN(C)C(C2(CF)CC2)=O)C)=O)nccc(Br)c1O 13479,c1(C(N(CCCCN(C(=O)CCc2ccn(C)c2)C)C)=O)csc(C(C)(F)F)n1 13480,C1(CC)(OCCC(=O)NCCN(C)C(C2CCN(C)C2)=O)CC(C)(C)C1 13481,C(C(CC(C)C)C(=O)NCC(C)CNC(c1nccn2cnnc12)=O)OC 13482,C1(C)(C(=O)NCC2CN(C(CS(=O)(=O)NCC)=O)CC2C)CCC2CC2C1 13483,N(C(=NCc1cc(C(F)(F)F)nn1C)NCc1nnc(C2CC2)s1)C(COC)C 13484,c1(OC)ccc(C(=O)N(CCCN(C(=O)C(F)(F)c2cnn(C)c2)C)C)c(C)n1 13485,CC(C)C(C#N)C(=O)N1CCC(NC(c2cnc(-c3cnccn3)s2)=O)C12CC2 13486,c1(C(=O)NC23CC(C(N(C4(C#C)CC4)C)=O)(C2)C3)cccc(O)c1 13487,CC#Cc1ccc(C(N2CCN(C3CC3)C(C#N)C2)C(=O)NC2CC2)cc1 13488,C(CC1=CCCCC1)N(C(c1cc(Cl)cs1)C(=O)NCC(C)C)C 13489,N1(C(c2cnc(C)c(Cl)c2)=O)CC2CC1CCN2C(C1CCSC1)=O 13490,c1(C(N2CCC(N(C)C(c3ccccn3)=O)C2)=O)ccc(C(C)(F)F)nc1 13491,N1(C(CCN(C)CC)=O)CCC(C)N(C(=O)CCCCC(N)=O)CC1 13492,O=C(C1=CCCSC1)NCCCCCCNC(C1COCCC1c1ccccc1)=O 13493,C1(C(N(CCNC(C2(C3CCC3)CC2)=O)CC)=O)CCCCN1C(C)=O 13494,c1(C(N(C)CCOCCNC(C2CCC23CCC3)=O)=O)cc2cccnc2cn1 13495,C1(C(=O)NCc2nc(CC)[nH]n2)C=CCN(C(C2CCCC(=O)C2)=O)C1 13496,N1(C(C(C=C)C)=O)CCN2CCN(C(c3cc(Cl)c[nH]3)=O)CC2C1 13497,N1(C(C(C)(C)CC(F)F)=O)CCN2CCN(C(=O)C3=CC4CCC(C3)C4)CC2C1 13498,C1(CCNC(Cc2c(C)n[nH]c2C)=O)CN(C(c2nn(C)cc2Cl)=O)CC(C)O1 13499,C1(N(C)C(C2CC2(C)C)=O)CN(C(=O)Cc2ccc(Cl)cn2)CC1(C)C 13500,c1(C(=O)NC2CCN(C(CC=CCC)=O)C2C(C)(C)C)ncnc2c1CCC2 13501,c1(C(=O)NC(C2CCN(C(=O)C(C)CC(C)(C)C)C2)C)ccc2nncn2c1 13502,c1(C(C)NC(CS(CC)(=O)=O)=O)ccc2c(c1)CN(C(=O)C(C)C(F)F)C2 13503,N1(C(Cc2n(C)nnc2)=O)CCC=CC1C(N1CCOC(CC(N)=O)C1)=O 13504,N1(C(N(c2ccc(C)c(C)c2)C)=O)CCCc2ccc(Br)cc2C1 13505,CN1CC=C(C(=O)NCCC(c2ccccc2)N(C)C(C2CC3(CSC3)C2)=O)C1 13506,c1(C(N2CC(C(N)=O)(CNC(C(C)n3cncn3)=O)C2)=O)ccnc2[nH]ncc12 13507,c1(OC)ccc(-c2cncc(C(=O)N(C)CCN(C)C(C3CC3Cl)=O)c2)c(C)c1 13508,Cc1[nH]nc(Cl)c1C(=O)NCC1CC(NC(=O)Cc2cccnc2)CC1O 13509,N1(C(C(CC)(CC)CO)=O)CCOC2(CCCN(C(=O)CCC(=O)OC)C2)C1 13510,c1(C(C)C)ccc(C2CCN(C(=O)CN3CCCCC3)CC2)cc1 13511,c1(C(=O)NC2C(NC(CCC=C)=O)C2)ccc(NC=O)cc1.C1CCN1 13512,Cc1cc(=NC(C)CCC2CCCCC2)[nH]c(=NCC=CBr)[nH]1 13513,c1(C(=O)NC2CC(CNC(C3=CCCC3C)=O)C2)n[nH]c2c1CCSC2 13514,C1(C(=O)NCC2(C)CC(NC(CC3(OC)CC3)=O)C2)CC(c2ccccc2)=NO1 13515,c1(C(N2C(CNC(COCCCOC)=O)COCC2)=O)cc2ccccc2s1 13516,N1(C(C2CCSCC2)C(=O)NC(C(=O)OC)C)C2CCC1CC(CO)C2 13517,C1(NC(C(N2CCC(C)(CCO)C2)c2ccc(CF)cc2)=O)CCC(F)(F)CC1 13518,CC(C)(O)C(C)(C)C(=O)N1CCCC1CNC(C1OCC2CCCC12)=O 13519,C1(C)(OCC(=O)NCC2(CN(C(=O)CCCc3nncn3C)C)CC2)CCCC1 13520,C(=O)(CC(CC(C)C)NC(c1csc(C)c1)=O)NC(C#CCC)(C)C 13521,c1(C(=O)NCCC(C)(C)NC(CC(C)C(F)F)=O)cc2nccc(Cl)c2s1 13522,C(=O)(C#Cc1ccccc1)N1CC2C(C(=O)Nc3cc(OC)ncc3Br)C2C1 13523,C1(CNC(CCN(C(C2(C(C)C)CCCC2)=O)CC)=O)CC(C)CC(C)C1 13524,CC#CCC(C)NC(C1(CCNC(=O)CC(Cl)Cl)CC1)=O 13525,c1(C(=O)NC2CC(CNC(C3C(C)CC(=O)N3)=O)C2)cc(O)ccc1[N+](=O)[O-] 13526,c1(C(N2CC(NC(=O)C(F)C3CCC3)(CO)C2)=O)cncc([N+](=O)[O-])c1 13527,C1(C(F)(F)F)(C(N2CCOCC2)=O)CC2CC2C1.C12(CO)CN(C1)C2.O=C1CN1 13528,C1(C(=O)NC2CC(NC(c3c(C)n[nH]c3)=O)CC2O)C(F)(F)C12CCC2 13529,c1(NCC(N2CC3CN(C(=O)COCC4CC4)C3C2)=O)ccc2c(c1)OCO2 13530,C(C1=CCCOC1)NC(C(c1cccs1)NC(c1cc(CO)on1)=O)=O 13531,N1(C(C=C(C)C)=O)C2CCC1C(CNC(=O)C(F)F)C2 13532,Cn1ccc(C(N2CC(=C(F)CNC(c3ccsc3)=O)C2)=O)c1C1CCC1 13533,C(C)(C)(CCN(C)C(c1cnc(C(C)(C)CF)o1)=O)NC(C1CC(OC)C1)=O 13534,c1(C(=O)NC2CC(F)(CNC(C(C)C3CCOC3)=O)C2)[nH]nc([N+](=O)[O-])c1Cl 13535,CC1C(NC(=O)CN2C(=O)CCC2=O)CCN1C(=O)Cc1ccccc1Cl 13536,N1(C(C2C(NCc3n(C(C)(C)C)ncc3)C2)=O)CCSC(C(N)=O)C1 13537,C#CC1(OC)CC2CCCC12.C12CN(CCO1)C(=O)C1CCC1(OC)NC2=O 13538,C12(CNC(CCNC(=O)CO)=O)CC1CN(C(c1cc(-n3cccc3)ccn1)=O)C2 13539,C(=O)(C(CC(C)C)N(C)C)N(C(C(=O)NCc1c(C)c[nH]n1)C1CC1)C 13540,N1(C(c2c(CC)n[nH]c2)=O)CC2CC2(CNC(=O)C(O)CC2CC2)C1 13541,n1(CC)cc(S(=O)(=O)NCC2CCCC2C)cn1 13542,N1(C(Cc2c(C)nc[nH]2)=O)CC2CCCC1C2CNC(c1cn[nH]c1)=O 13543,N1(C(C(CC)O)=O)CCCC(N(C)C(c2ccnc(OC)c2)=O)C1 13544,CCCCCC(C)CC(=O)N(C1CC(NC(C2C=CCS2)=O)C1)C 13545,C(=O)(CC(C)(C)O)N1CC(C(C(N2CC(N(CC(C)C)C)C2)=O)O)C1 13546,Cc1cc(CCNC(=O)C(Cn2cncn2)NC(=O)CC2CCSC2)n[nH]1 13547,C(=O)(C(CC(C)C)NOC(=O)C(C1(O)CCCCC1)(F)F)OC 13548,C1(C(=O)OC(C(C)C)C(N2CCCc3ccccc32)=O)CCc2cnccc2N1 13549,C(CCC(=O)NCC1CC2(CC2)C(=O)O1)(C(=O)O)N(C)C 13550,c1(C(N2CCC(O)(C(C)NC(c3cc(C(N)=O)no3)=O)C2)=O)ccc(Cl)nc1Cl 13551,C(=O)(CCC(=O)N1CCC(C(C)(O)CNC(=O)C(C)SC2CC2)CC1)NC 13552,C1(CNC(C2CSCCS2)=O)CCCN(c2nc(C3CCCC3)ns2)C1 13553,C1(C)(C(=O)NCC(N2CCCCC2)C)CN(C(=O)C=CCN2CCC2)C(C)(C)C1 13554,C1(N)(C(=O)Nc2cc(COC)c(OC)cc2)CCC(C)(C)CC1 13555,CC1CCC(NC(c2nn[nH]c2Cl)=O)CN1C(=O)CCCCc1ccccc1 13556,c1(OC)ccc(C(=O)NCC2(C)CCCN2C(c2cnc(S)n2C)=O)c(N)c1 13557,CN1CCN(C(=O)C(CC(F)F)NC(C2CC3CCCC3C2)=O)CC1=O 13558,N1(C(C(CC(=C)C)C)=O)C2CCC1CC(N(C)C(c1ccc(Br)s1)=O)C2 13559,c1(C(C(=O)NCCCOCCN(C)C(c2cnc(O)s2)=O)O)ccc(Cl)cc1 13560,c1(C(=O)NC2C(C(=O)NCC3CCC3)CCCC2)cc(Br)cc([N+](=O)[O-])c1Cl 13561,CCC(CC(=O)NCC1(NC(C2CCCSC2C)=O)CCC1)c1ccccc1 13562,c1(C(N2CCC(NC(=O)C=Cc3cocn3)CC2)=O)ccc(Br)cc1[N+](=O)[O-] 13563,C1(C(=O)NC(C2CCN(C(Cc3c(C)nc(C)s3)=O)C2)C)CCCCC12CCC2 13564,C(=O)(C1CCCc2ncccc21)N(CCCN(C)C(C1CC2(CCC2O)C1)=O)C 13565,c1(NC(C2CCN(Cc3cccc(-c4nn[nH]n4)c3)C2)=O)cc(Br)ccc1Br 13566,C1(NC(c2cc(Cl)cnn2)=O)C2CCC1N(C(=O)Cc1cccc(F)c1O)C2 13567,N1(C(CSCC=C)=O)CCN(C(c2cnn(C)c2C(C)C)=O)CC1CC(F)F 13568,N1(C(CC2(CSC)CC2)=O)CC(NC(=O)C(C)C(C)O)CC12CCCC2 13569,c1(C(C)(C)C)cccc(C(=O)NC2CCC(CNC(=O)CCc3cscn3)C2)n1 13570,C1(NC(C(CCC)C)=O)COC2(CCN(C(c3ccc(CC(C)C)cc3)=O)C2)C1 13571,N1(C(C2CC(CNC(CCCN(C)C)=O)C2)=O)CCCC(F)(CO)C1 13572,C1(NC(C(CC)(C)OC)=O)CCCCN(C(c2ccc(C)nc2N)=O)C1 13573,CONC(=O)C(=O)N1CC(F)CC1CN(C(=O)CSCC(N)=O)C 13574,N1(C(CC=C=C)=O)CC2CC(NC(c3csc(Cc4ccc(F)cc4)n3)=O)C1C2 13575,N1(C(c2cn(C)nc2)=O)CCC(CNC(c2ccc3n[nH]cc3n2)=O)C12CCC2 13576,N1(C(C(CO)NC(C)=O)=O)CCn2nc(C(=O)NCC(O)CO)cc2C1 13577,N1(C(CCC(C)OC)=O)CCC(NC(=O)CSc2ccncc2)C(F)C1 13578,CC(CF)CC(=O)NCC1CC1CNC(c1cc(-c2ccncc2)ccn1)=O 13579,N1(C(c2c(C)nc(C(C)C)s2)=O)CC2(CCC2NC(C2COC(C)(C)CO2)=O)C1 13580,c1(C(=O)NC2CCC(CNC(C(C)=C3CC3)=O)C2)cnn2c1C(C)CCC2 13581,c1(C(N(C2CCCC2)CCCNC(C2C(C)(C)CC2)=O)=O)cc[n+]([O-])cc1 13582,c1(C(=O)NCC2C=CCN2C(=O)CC2CCCOCC2)ccc(F)cc1Br 13583,C(N=c1[nH]c2c(c(=NCC3(C4CC4)CC3)[nH]1)COC2)c1cc(Cl)cc(Br)c1 13584,n1(C(C)C)ccc(C(=O)NC(C)(C)C(=O)NC(C2CCC2)C)n1 13585,CC12COCC1CN(C(N1CCCC1C(O)C(F)F)=O)C2 13586,c1(C(=O)NC2C(NC(CC(=O)NCC)=O)CCC2)cccc(C)c1Br 13587,N1(C(CSCCC)=O)CCN(C(=O)C(C)Cc2ccc(Cl)cc2)C(C2CCC2)C1 13588,C1(SCC)CCCC(N=c2[nH]c(=NCc3cc(O)n[nH]3)[nH]c3ncn(C)c23)C1 13589,c1(C(=O)NC(CC)CN(C(=O)CSCc2cccnc2)C)cn(C)nc1C(C)C 13590,C1(NC(C(C)C=Cc2ccccc2)=O)CN(C(=O)CCCC2CCC2)CCC1C 13591,Cc1nn(C)c(F)c1C(=O)NCCN(C(=O)Cn1ccc(C(F)(F)F)n1)C 13592,Cn1nc(CNC(C2CCCCC2)=O)cc1NCCC(O)C(F)F 13593,C1(N2CC(C(=O)NCC3C(NC(=O)COCCF)CC3)C2)CCCCC1 13594,N1(C(c2n(COC)ncc2)=O)CCC(C)C(CNC(c2nc(Cl)cs2)=O)C1 13595,N1(C(c2c(C)ccnn2)=O)CC2(CC(NC(C34CC3COC4(C)C)=O)C2)C1 13596,c1(C(N2CCC(N(C(c3nn(CC)cc3Cl)=O)CC)C2)=O)cc2n(n1)CCC2 13597,Cc1cccc(C(N2CC(O)(CNC(c3ncccc3N)=O)C2)=O)c1C 13598,c1(OC)[nH]c(=NC2CCCCCN(C(=O)C(=O)NC(C)C)C2)sc1C 13599,C1(CNC(C2N(CC)CCCC2)=O)CN(C(C2(CC3CC3)CC2)=O)CC12CCC2 13600,N1(C(C2(C(=O)OC)CC2C)=O)CC2CCCN(C(=O)C(C(C)C)NC(N)=O)C2C1 13601,CC(CCCC(=O)NCc1cccc(CO)c1)NC(c1cccc(CC#N)c1)=O 13602,C1(C)(C(=O)NCC2CC(NC(C3CC(C(=O)OC)C3)=O)C2)CCCNS1(=O)=O 13603,c1(N(C(=O)OC(C)(C)C)C2CC2)cnn(C)c1.C1(=O)CCN(C)CC1=O 13604,c1(CCC)[nH]ccc1C(=O)N(C1(CC(=O)NC2(CC(C)C)CC2)CC1)C 13605,c1(C(C(N2C(CNC(c3cc(I)on3)=O)CC2)=O)F)ccc(C(F)(F)F)cc1 13606,Cc1csc(=O)n1CCC(=O)N(C)CCN(C(=O)C=CC(=O)N(C)C)C(C)C 13607,C1(C(=O)NCC2OCCN(Cc3nc(CCC)on3)C2)Cc2ccccc2O1 13608,N1(C(C2C3CCCC23)=O)CC2C(Cc3cn(CCC(F)(F)Cl)nn3)C2C1 13609,C1(N(C(C2CSC2)=O)CC)CCCN(C(c2ccc(O)c(Cl)c2)=O)CC1 13610,c1(CC)ncc(C(=O)NC(CNC(C2CC3C=CC2O3)=O)CCOC)c(O)n1 13611,C1(C(N2CCCCC2)=O)CCCN(C(=O)CN(C2CC2C(F)(F)F)CC2CCC2)C1 13612,C1(OC(C)=O)CCCN(C(=O)NC(CO)C(C)OC(C)(C)C)C1 13613,Cc1cc(C(=O)N(C)CC2CCN(C(=O)C#CC(=O)N(C)C)CC2)ccn1 13614,C1(N(C(=O)C=CC2CCCO2)C)CCCN(C(C2CCOCC2)=O)CC1 13615,C1(OC)CCC12CC(C(=O)NC1CC(CNC(=O)C3=CCCSC3)C1)C2 13616,c1(C(N2CCC(C(C)C(=O)NCC(C)(C)O)CC2)=O)ccc(C#N)cn1 13617,c1(C(=O)NCC(C)NC(C2C(OCC)C2C)=O)cnc2c(c1)nnn2C 13618,n12nc(cc1C)C(=O)NCCOCCCNC(=O)C2.C12(CC1)N(C)C2=O.CC 13619,Cc1coc(C)c1CNC(=O)C(C)N(C(c1ccccc1)=O)C1CC1 13620,N1(CCNC(C(C2CN(C(=O)C=Cc3ccco3)C2)OC)=O)CC2CC2C1 13621,c1(OC)cnc(Br)cc1C(N1CCN(Cc2cnn(C)c2)CC1CC#N)=O 13622,C1(C(N2CC(O)(CNC(c3c(C)cc[nH]3)=O)C2)=O)C2C(=O)OCC12Br 13623,c1(CC(=O)NC2CC(NC(=O)C(F)=CC3CC3)C2)noc2ccccc12 13624,Cc1cc(C(=O)NC2CCCC(NC(C3C4CCCOC34)=O)C2)cc2ccsc12 13625,C(c1ccccc1)=C(C)C(N1CC2CC2(C(=O)NC(C)(C)C(F)(F)F)C1)=O 13626,C1(C(=O)Nc2cccc(NC(C(CC)=CC)=O)c2)CC(=O)c2ccccc2C1 13627,C#Cc1ccc(NC(C2CC(F)(F)CN2c2cc(C(F)(F)F)ncn2)=O)cc1Cl 13628,C1(C(C)C#N)CCN(C(=O)CCC2CCC(NC(=O)COC3CCC3)C2)CC1 13629,CN1CCC(CCC(=O)NCCC2CCCN2C(c2cc(C3CC3)on2)=O)CC1 13630,N1(C(CCNC(=O)OC)=O)CC2CC(C(=O)N(c3ccccc3OC)C)C(C2)C1 13631,C1(CN(CC(C)C)C(c2cn(CCOCC)nc2)=O)CCCC12CC2 13632,C1(NC(Cn2ncn(C)c2=O)=O)CCN(c2cc(C(F)F)ncn2)CC1O 13633,C(=O)(C(C)(CC)CCC)NCCCNC(C1(CC#C)CCC1)=O 13634,n1(CCC)cc(C(=O)NCC(O)CN(C(=O)COCc2ccccc2)C)c(C)n1 13635,C(=O)(CCC(=O)NCC(=O)NC1CCC(NC(CC)=O)C1)N1CC(C(C)OC)C1 13636,C=C1CC2(C1)CN(C(=O)C(CC(C)C)N(C(=O)CCC1CC1(F)F)C)C2 13637,C1(C(=O)NC2(C(C)C)CCC2)CCC2(CC2)N1C(c1cnc(O)o1)=O 13638,c1(C(=O)NC2C(NC(c3cccc(CC)c3)=O)CCCC2)cc(Cl)cc(F)c1N 13639,C1(C)(CC)NC(=O)N(CC(=O)NCCNc2ccc(Cl)cc2CO)C1=O 13640,c1(NC(=O)C(F)OC(F)(F)F)cn(CC(=O)NOCC2CCNCC2)nn1 13641,CCC(CC(C)C)C(=O)N1CCC(C(C)NC(c2ccc(O)c(CO)c2)=O)CC1 13642,CC1CCC(C(=O)N(C)Cc2nnnn2C)N1C(c1ccn(C)n1)=O 13643,N1(C(c2[nH]c(=NC)sc2)=O)CC(N(C(=O)C(C)SC(C)C)C)C(C)(C)C1 13644,C=CCCCC(C)NC(=O)C(C)CNC(=O)CN(C)C(=O)OC 13645,Cc1cc(C(=O)NCC2CC(NC(C3(CO)CC3)=O)C2)n(C2CCC2)n1 13646,CCCC(C(=O)N1CC(N(C)C(C2(C3CCCO3)CCOCC2)=O)C1)OCC 13647,c1(C(=O)OC)c(F)ccc(CN2CC(F)CC2c2cccc3c2OCO3)c1F 13648,N1(C(C2(C(=O)NC)CC2)=O)CCCC(O)(CNC(=O)C(C)CN(C)C)CC1 13649,Cc1cc(NC(c2ccc(CNC(c3cnns3)=O)s2)=O)c(O)cc1F 13650,c1(CC)ccnc(CNC(=O)CC2CC(NC(c3cc(OC)ccn3)=O)C2)c1 13651,C12(CNC(C3C(OC)C3)=O)CC1CN(C(C1CCN(C(=O)C(C)(C)C)CC1)=O)C2 13652,N1(C(CCC(C)C)=O)CCCC2C1CCCCN2C(=O)CCc1cccn1C 13653,C(=O)(C(F)C(F)(F)F)N(C1CCN(c2cc(CC)ncn2)CC1)Cc1ccccc1 13654,N1(S(=O)(=O)CC2CC2)CCCC2C1CCN2Cc1cc2ccncc2[nH]1 13655,C12(CNC(C=CC(C)(C)C)=O)CCC(CC1)CN2C(C1CC12CCC2)=O 13656,N1(C(CC(=O)OC)=O)CC(C(=O)Nc2c(CO)noc2C)CC12CCC2 13657,C1(CC)C(C(=O)NCC(O)CC2CCCC2)CCN1C(c1ccncc1CC)=O 13658,CC1=C(C(=O)N2CC(CNC(=O)CN3CCSCC3)CC(C)C2)CCCO1 13659,CCC(CC(=O)N1CC2CN(C(c3c[nH]c(=NC)o3)=O)CC2C1)C(C)C 13660,N1(C(=O)CC2CCC3CC3C2)CC23CCCC2(C1)CN(C(C1CCC=CO1)=O)C3 13661,C1(CNC(Cc2nccc(C)c2)=O)C(C)CCCN1C(c1ccc(C)cc1F)=O 13662,C(C(C)(C(C)C)C(C)C)NC(CC1C(C)CN(C(c2sccc2Cl)=O)C1)=O 13663,c1(C(=O)NC2CN(C(c3ccn(C)c3)=O)C3C2C3)ccc2cc[nH]c2n1 13664,c1(OC)cc(C(=O)NC2CCC(NC(=O)Cn3cc(Cl)cn3)CC2)ccc1[N+](=O)[O-] 13665,c1(C(N(CCNC(C(N)=O)=O)C2CC2)=O)cc2c(O)ncnc2cn1 13666,c1(CC)nccnc1C(N1CCCCC1CCN(C)C(C1(C)CCC(=O)N1)=O)=O 13667,C(C(C)(C)C(=O)N1COC(C)C1)N(C)C.C12(C)CCCN1C(=O)C(C)(C)NC2C 13668,c1(C(N(C(CNC(C2CN(C(C)=O)C2)=O)C)C2CC2)=O)ccc(C)c(Br)c1 13669,Cc1ccc(C#N)cc1C(N1CC2CC1CCC2NC(=O)C(F)(F)C(F)F)=O 13670,C1(NC(c2c(F)ccnc2F)=O)CCN(C(=O)CCc2cc[nH]n2)CCC1CO 13671,Cc1conc1CC(=O)N(CC(=O)N(C)Cc1cccnc1)CCO 13672,N1(C(CC2CC(OC)C2)=O)CC(CC(N2CCCC(CCF)C2)=O)CC1C 13673,c1(C(N(C(C)CCNC(C2SC3C=CC2CC3)=O)C)=O)cc2ccc(Cl)cc2s1 13674,c1(CCC)cc(C(=O)NC2CCCCC2NC(=O)CC2CC(C)(C)C2)cc(O)n1 13675,c1(C(C)=O)ccccc1OCCC(=O)NCC1CCCCN1C(=O)C(C)CCO 13676,c1(SC)cccc(C(=O)NCCN(C(c2cnc(S)[nH]2)=O)C2CC2)c1 13677,c1(SCCC(=O)NC(CN(C(CNS(NC)(=O)=O)=O)C)C)ccccc1Cl 13678,Fc1ccc(F)c(NCC2CCCC(C(F)(F)F)C2)c1F 13679,C(=O)(C(C)(C)C(N)=O)NCCC1C(C)CN(C(=O)COCc2cccnc2)C1 13680,c1(NC(C2C(C(=O)OC)C2)=O)ccc(C(=O)Nc2cnc(O)cc2C)cc1C 13681,Cc1cc(C(=O)N(C2CCCN(C(C3CNC(=O)C3)=O)C2)C)cc([N+](=O)[O-])c1O 13682,c1(OC)ccc(CC(=O)NC2CC(C)(NC(=O)CCc3ccccn3)C2)cn1 13683,C(=O)(C1=CCCOCC1)NC(C(=O)N(CC(C1CC1)OC)C)C1CCOC1 13684,C1(CC(=O)NC(CNC(c2scc(C)c2)=O)CO)CCCN(C(C)C)C1 13685,C(=O)(C(C)(C)CN(C(=O)C(CC)n1cncn1)C)NCC(CCC)OCC 13686,n1(CC(C)NCCCC(C)(C)CO)cnc2c(cnn2C)c1=O 13687,N1(C(c2c(CC)c[nH]n2)=O)CCC2C(C(=O)NC(c3noc(C)n3)CC)C2C1 13688,CN1C(=O)Cc2ccc(C(=O)NC3CC3CNC(=O)C=Cc3cccn3C)cc21 13689,CCCCCCCC(=O)N1CCC(N(C)C(c2cccc(-c3nccs3)c2)=O)C1 13690,C(=O)(C(C)CCCC)N1CC(CC(=O)NCC=CC)OCC1 13691,CCCC(O)(CNC(=O)N(C(c1cccc(C)c1)CO)C)CCC 13692,N1(C(Cc2c(C)non2)=O)CC(NC(=O)CCC2CCCC2)CCC1C 13693,C=CC(F)(F)C(=O)N(CCCNC(=O)C(=O)NC1CC1)C(C)C 13694,c1(C(=O)NC2(CNC(Cc3cn(C(C)C)nc3)=O)CC2)ccc2[nH]c(=N)sc2c1 13695,C1(CNC(c2n(C)c(O)nc2)=O)COCCN(C(c2csc(C#N)c2)=O)C1 13696,c1(OCC(=O)OC2CN(C(COCCC=C)=O)C2)ccc(OC)cc1Br 13697,C1(CC(=O)N(C2CC2)CC2N(C(C(C)Cn3ccnc3)=O)CCC2)CC2(CCC2)C1 13698,N1(C(CCCNC(N)=O)=O)CCOCC(C(N2CCN(CCO)C(=O)C2)=O)C1 13699,Cc1nc(C(F)(F)F)c(N(C2CCCN(C(c3ccco3)=O)C2)CCO)o1 13700,C1(CC#C)(C(=O)NCC(c2cccc(Br)c2)C)CCCNC1 13701,N1(C(C(C)C2CC2)=O)CC(C(=O)NCc2ccnc(F)c2F)C2(CCC2)C1 13702,N1(C(=O)OCc2ccccc2)CCc2nc(CNC3CCC=C3Br)cn2CC1 13703,c1(C(=O)NCC2(C(=O)NC(COC)C(N)=O)CC(=C)C2)cnc(C)n1C 13704,Cc1cc(C)c(C(N2CCN(C(c3ccns3)=O)CC2C(C)C)=O)cc1N 13705,Cc1cc(CC(=O)NC(CNC(=O)Cc2[nH]cnc2C)C(C)(C)C)n(C)n1 13706,C1(C2CCCC2)(C(N(CC(CNC(c2c(OC)c[nH]n2)=O)C)C)=O)CCNC1=O 13707,C1(CNC(C(C=C)C)=O)CN(C(=O)Cc2csnn2)CC12CC2 13708,O=C1CCC(S(=O)(=O)N(CCO)CC2CCCN(C(=O)C3=COCCC3)C2)CC1 13709,Cc1nnc2n1CC(CNC(=O)CCn1cncc(Br)c1=O)CC2 13710,C1(CC)CC(C(N2CC(NC(c3cc(C(F)F)cc(F)c3)=O)C2)=O)CC(=O)N1 13711,Cc1cc(C(=O)NCC2(O)CCCN(C(c3cc(C(F)F)cs3)=O)C2)cnc1O 13712,C12(CNC(CC3C(CC)C3)=O)CC(NC(c3scnc3Br)=O)(C1)C2 13713,C(c1cccc([N+](=O)[O-])c1)=CC(=O)NC1(C)CCN(C(C2(O)CCOC2)=O)C1 13714,c1(C(C(n2cc(C(C(=O)OC)(C)C)nn2)C)NC2CC3CC3C2)cccc(Cl)c1 13715,c1(OC(C(C)N(C(=O)C=CC(F)(F)F)CC)C)sccc1C(=O)O 13716,N1(C(c2c(C#C)c[nH]n2)=O)CC(C)C(NC(c2ccc(=O)oc2)=O)C(C)C1 13717,N1(C(CCCc2onc(C(C)C)n2)=O)CCN(C(C2CCC(O)C2)=O)C(C)C1 13718,C1(CNC(C2CC(C#C)(O)C2)=O)CN(C)CCN1C(C1CC(C)C1)=O 13719,C(C(CC(=O)NC1CCN(C(=O)Cc2ccn(C(F)F)n2)C1)C(F)(F)F)N(C)C 13720,Cc1cc(Cl)cnc1S(=O)(=O)N1CCSC(c2cnn(C(C)C)c2)C1 13721,c12ccnc(n1)C(=O)N(C1CCC(C)CC1)C1CCN2C1.CC.SC 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13846,C1(C(N2C(C(C)NC(c3c(C)cc(C)nc3)=O)CCC2)=O)CC(C(C)(C)C)=NO1 13847,N1(CCC)CCCCC1C(=O)NCCC(C(C)C)NC(=O)Cc1cc(C)[nH]n1 13848,C1(C)(C(=O)NCC(CN(c2nc(C)cc(C(=O)NC)n2)C)C)CCC(C)=C(C)C1 13849,c1(C(=O)NC(CNC(c2cc(SCC)ncc2)=O)CC)ncnc2ccsc12 13850,c1(OC)cc(C(=O)Nc2cccc(CN(C)C)c2)cnc1-c1sccc1CO 13851,c1(C(=O)NCC(CO)NC(c2ccn(C)c2)=O)cccc(S(C)(=O)=O)c1 13852,C1(CNC(C(C(C)C)OC)=O)(NC(=O)C(c2cccnc2)C)CCC(F)(F)CC1 13853,CC1CCN(C(=O)CSC2CC2)CCN1C(C12CC(CO)(C1)OC2(C)C)=O 13854,CC12CC(C(=O)NCC3CC3NC(c3cc(CO)[nH]n3)=O)(CCO1)C2 13855,N1(C(CS(CC)=O)=O)CCC2(CCCC2NC(=O)CCSc2n[nH]c(C)n2)CC1 13856,c1(N(C2CN(C(c3c[nH]cc3Br)=O)C2)C)cc(Cl)nc(CS(C)(=O)=O)n1 13857,N1(C(COCC(=C)C)=O)CCC(CNC(C2CCS(=O)(=O)C2)=O)C12CC2 13858,N1(C(C2CC(C)OC2C)=O)CCC(C2(CNC(=O)C3CC3)CCOCC2)CC1 13859,c1(CC)nc(C)c(CC(=O)NC2CC3(C2)CC(NC(C2CC2F)=O)C3)c(C)n1 13860,N1(C(C=C(COC)C)=O)CC(NC(=O)C(F)CC2CCCC2)C(C)(C)C1 13861,N1(C(c2cc(C)sn2)=O)CCC(O)(CCNC(C2(CO)CCOC2)=O)C1 13862,N(C(=NCCCOC(F)F)NCc1ccc(OC(F)F)cn1)CC1C(C)CCC1 13863,C1(C(N2CC3C(CNC(c4c(C)cccc4C)=O)C3C2)=O)CCC2CCCCN12 13864,c1(CC(=O)NCCN(C(=O)CC2CCNC2=O)C)cc(Cl)sc1Cl 13865,N1(C(CC2CC(CC)C2)=O)CCCC(CCNC(C2CC(OC)C2)=O)CC1 13866,C(=O)(C(C)CS(C)(=O)=O)N(CCNC(C(C1CCC(C)CC1)CC)=O)CC 13867,C1(NC(N2CC3C(CC#N)CC(C3)C2)=O)CCCC12CCOCC2 13868,C#Cc1cc(NC(C2CC(=O)C2C)=O)ccc1C 13869,N1(C(C2C(OC)CCC2)=O)CCC(C)(C(=O)NCC2(C)CC(C)=NO2)C1 13870,C1(NC(c2cc(CCOCC)on2)=O)CC(F)CN(C(=O)COCCOC)C1 13871,CCCCC(CC)CCC(=O)NC(C)(CNC(C1CCC1C(C)(C)C)=O)C1CCC1 13872,N1(CCC(C)NC(=O)C=CC(F)F)CCCC(C)C1 13873,N1(CCC(=O)NC(C2CCCN2C(c2nncs2)=O)(C)C)CCP(C)(=O)CC1 13874,c1(C(=O)NCC2CC(C)N(C(C3C(C)(C)OC3(C)C)=O)C2)ncsc1S(N)(=O)=O 13875,N1(CCS(CC)(=O)=O)CCC(c2ncc(C(=O)O)s2)C1 13876,C1(C2(O)CCN(C)CC2)(C(=O)NC(CCCNC(c2c(C)occ2)=O)(C)C)CC1 13877,C(C)(C)(C(O)C(F)F)N(C(=O)Nc1c(C)nn(-c2ccc(F)cc2)c1)C1CC1 13878,Cc1nc2[nH]c(C(=O)NCCCCN(C)C(C3(C)CC4CC4C3)=O)cc2s1 13879,c1(-c2onc(Cc3ncc(C)cc3Br)n2)noc2c1COCC2 13880,C12(C(=O)NC(CC(=O)OC)C)CCC(n3cc(CN(C)C(=O)NC)nn3)(CC1)C2 13881,Cc1cc(C(N2CCN(C(=O)Cc3cnn(C)c3)C(CC(F)F)C2)=O)cc(O)n1 13882,N1(C(C2(C3CC4CCC3O4)CC2)=O)CCC(F)(c2cn(C(CF)C(F)(F)F)nn2)C1 13883,c1(CC)noc(CN(CCNC(=O)CCc2nc(C)no2)C2CC2)n1 13884,c1(-c2nc(CCCN(C)C)nn2CC(C)(C)C)cncc2c(Cl)cccc12 13885,c1(C(N2CCCC(C(C)NC(C(C)=C3CC3)=O)C2)=O)cc2cc(C)c(C)cc2o1 13886,N#CC12CCC(CN3CC(c4ncccn4)C3)(CC1)CC2 13887,c1(-n2ccc(C)n2)cccc(C(=O)NCCC2(O)CCOC2)c1 13888,C1(NC(CC(CC)OC)=O)CN(C(c2nccc(C(F)(F)F)n2)=O)C(C)(C)C1 13889,N1(C(c2nncc(C)c2)=O)CCC(C)C(NC(c2cc(C)sc2C)=O)C1 13890,CC1C(C(=O)N(C)Cc2ccnn2C)CCN1C(C1CCCC1)=O 13891,N1(C(CC2C(NC(C(F)=CCC)=O)CC2O)=O)CCCC2C(O)CC12 13892,Cc1nn(-c2cccc(Cl)c2)c(C)c1CN(C1(CCO)CCCC1)C 13893,c1(CC(=O)NC2CCC(C)(CNC(C3(COC)CC3)=O)C2)c(Cl)ccc(O)c1Cl 13894,N1(C(c2n(C(CC)C)ncc2)=O)CC(NC(c2cnc(O)c(F)c2)=O)C2(CC2)C1 13895,N1(C(C2N(C=O)CCC2)=O)CCC(C=CC(=O)O)CC1.C1CN1C1CC1 13896,c1(OC)cc(C(=O)N(C(CNC(=O)C(C)=C(C)C)C2CC2)C)[nH]n1 13897,c1(C(=O)NCC23CCC(NC(C(C)SC(F)(F)F)=O)(C2)CO3)cc2nc[nH]c2cn1 13898,C(=O)(CC1=NN(C)C(=O)C1)N(CC(CC)OC)C.C1(=O)C(O)CN1 13899,C(=O)(CC(F)(F)C(C)C)N1CCCC(N(C(C(CCCOC)C)=O)C)C1 13900,N1(C(C(C2CCCC2)NC(C(CC2CCC2)OC)=O)=O)CC(C2CCCCC2)C1 13901,Cc1noc2nc(=NCC3CCn4ccnc4C3)[nH]c(N)c12 13902,C(=O)(C(F)CCC(C)C)N1CCCC(CCNC(C(CC)(F)F)=O)C1 13903,c1(C(=O)NCC(C)N(C(=O)CC(C)CF)CC)ccc(CO)c(F)c1 13904,c1(C(=O)NCCN(C(C(C(C)(C)C)SC)=O)C2CC2)ccc2c(c1)OCCC2 13905,N1(C(C(CCO)N(C)C)=O)CC2CCN(C(=O)CCn3cc(Br)cn3)C2C1 13906,C1(NC(C(C#C)(C)C)=O)CN(C(C2CC3(CC3)CO2)=O)CC1C=C 13907,C1(C(=O)NCCSCC)CC2(CC(NC(=O)CCC(=O)NC)C2)C1 13908,c1(C(C)(C)C)ccc(S(=O)(=O)N2CC3CC2CC3N2CCC(Cl)C2)cc1 13909,C1(C(=O)NC2C(CNC(CC(C)(C)OC)=O)CCCC2)CCC2(CC1)CC2(F)F 13910,C(=O)(N=c1cc[nH]cc1NCCCn1c(C)ncc1)C1(C(F)(F)F)CCOCC1 13911,C(CC1=CCCCC1)NC(c1c(CNC(C2(Cl)C(C(C)=O)C2)=O)ccs1)=O 13912,c1(C(N2CCN(C(C3CCSCC3)=O)C3CC23)=O)cc(Cl)c(F)cc1Cl 13913,C1(NC(c2c(C)nn(C(C)C)c2)=O)CCN(C(C2(C)CCC2)=O)CC1C 13914,C1(C)(C(N2CC3(C(NC(C=CCOC)=O)CC3)C2)=O)Oc2ccccc2NC1=O 13915,CC1CCc2[nH]c3ccc(C(N4CCN(C(=O)CCN(C)C)CC4)=O)cc3c2C1 13916,Cc1ccc(CNC(=O)C(C)(C)C2CCN(C(=O)C(C)OCC3CC3)C2)c(O)n1 13917,Cc1cc2ncn(CC(=O)NC(C)(C)CN(C)C(C3CC3(F)Cl)=O)c2cc1C 13918,c1(C(=O)NC2C(NC(CCc3cc(C)on3)=O)CC2)cn(C)nc1C(F)(F)F 13919,C1(C)(NC(c2c(CC)nccn2)=O)CCN(C(c2nccc(N)c2Cl)=O)CC1 13920,C1(C)(C(N(CC(CNC(C2C(OC)CCC2)=O)C)C)=O)CCC(=O)NC1 13921,N1(C(c2c(=N)[nH]cnc2)=O)CC2CCN(C(=O)COCCF)CC12 13922,N1(C(c2ccc(C(C)=O)o2)=O)CC=CC(C(=O)N(CC(C)C(C)C)C)C1 13923,N1(C(C2N(C(C)=O)CCC2)=O)CCC(C)C(CNC(=O)C(c2cscn2)N(C)C)C1 13924,C(=O)(CC1=NN(C)C(=O)C1)N1CCC(n2cc(CC=C)nn2)C(O)C1 13925,c1(C(N2CCC(C)C2CNC(=O)Cc2csc(S)n2)=O)cc(O)ccc1Cl 13926,c1(C(N2CC(C)(CNC(C3CC=CC3)=O)OCC2)=O)ccc(S(N)(=O)=O)cc1 13927,c1(COC)cnc(OC)c(C(=O)NCC#CCNC(c2coc(Cl)n2)=O)c1 13928,C1(c2n(CCC)nnn2)(NCC2(CC)CCCO2)CC(C)SC(C)C1 13929,C1(CNC(C2CC(SC)C2)=O)C=CCN1C(c1ncn(C)n1)=O 13930,N1(C(C23N(C(c4c(OC)ccs4)=O)CC(CO)(C2)C3)=O)CCCC12CCOC2 13931,c1(-n2cc(CN3C(CCCO)CCC3)nn2)cc(Br)ncc1Br 13932,N(C(=NCC(C)OC)NCC1CCCCC1)Cc1ccc(CC)cc1 13933,c1(CN2CC3C(C(=O)N(CCO)CCO)C3C2)cc(Cl)ccc1Br 13934,CC1(C)CC(CC(=O)NCC(C)(CO)NC(c2cccnn2)=O)C1 13935,c1(C(=O)OC)cc(F)cc2c1CCN(C(C1CCC(C(=O)N(C)C)O1)=O)C2 13936,C1(OC)CCN(CC(=O)NC2CCC(N(C)C(C3CC3(Cl)Cl)=O)C2)C1 13937,Cc1cnc(C=CC(=O)NCCC2COCCN2C(=O)Cc2cc(Cl)cs2)[nH]1 13938,N1(C(C=CC(=O)NC2CC2)=O)CCCCCC(NC(C2(C3CCC3)CC2)=O)C1 13939,C#CCCCC(C)C(=O)N(CCN(C(=O)CCc1cocn1)CC)CC 13940,C(c1ccccn1)=C(C(=O)N(CCOC)CCNC(C1CCOC1C)=O)C 13941,Cc1cc(C(N2CCN(C(=O)CC3=CCCC3)C(C)C2)=O)cc(F)c1C 13942,O=C1CC2C(C(=O)NCc3csc(CNC(c4c[nH]nc4Cl)=O)n3)C2C1 13943,C(=O)(C(C)C(C)(C)C)NC(C(C)C)CNC(=O)CC1CS(=O)(=O)C1 13944,N1(C(c2snnc2C)C(=O)NCC2(C(=O)OCC)CC2)CC2(CC2)CC1C 13945,CC1CC(C)(C(=O)NC2CCC2NC(c2cc(F)n(C)n2)=O)CCO1 13946,n1(CC(=O)NC(CC)CNC(c2cc(C(C)=O)cs2)=O)nc(C)cc1COC 13947,Cc1cc(=NCC2CN(C(c3cc(C(C)(C)C)on3)=O)CC2(C)C)c(C#N)c[nH]1 13948,c1(OCC)cncc(C(=O)N(CCCCCNC(c2cncc(OC)n2)=O)C)c1 13949,CCC(C)CCCC(=O)NC1CCCC1NC(c1c[nH]c(=N)o1)=O 13950,N1(C(CCC#C)=O)CC(NC(=O)CCc2cccnc2C)CC12CCCCC2 13951,C(CC(CC)C(=O)NC1CCCCC1C(=O)NC(C)CCOC)=CC 13952,c1(-c2ccc(N3CCN(C(c4ncc(OC)c(C)c4)=O)CC3)cc2)cc([N+](=O)[O-])nn1C 13953,C1(NC(C(c2cn(C)nc2)(F)F)=O)CCN(C(=O)CCOCC(F)(F)F)C1(C)C 13954,c1(CC)nc(C)c(C(=O)NCC(C(C)C)NC(=O)CCn2nc(C)cc2C)o1 13955,CN1CCC(C(N2CC3CC(C(=O)NC4CCN(CC5CC5)C4)(C3)C2)=O)CC1=O 13956,CCC(C)C(O)C(C)C(=O)N(CCC(=O)NCC1CC1)CCCO 13957,c1(C(=O)NCC2CCCCCN2C(=O)COC2CCCC2)cc2c(nn1)CCC2 13958,N1(C(C2CCC(N=[N+]=[N-])C2)=O)CCC2(CC1)CN(C(c1ccncc1)=O)CCO2 13959,Nc1nccn2ncc(C(=O)NC3CCC(CNC(=O)Cc4ncc(Cl)s4)C3)c12 13960,C1(C(=O)OCCOCC(C)(F)F)CCCCN1O 13961,CC1(C)CC(C(N2CCCC(CNC(C3CCC(=O)C3)=O)C2)=O)CC(C)(C)S1 13962,CC1CCCCC1C(=O)NCC1(CNC(=O)C(F)(F)c2ccncc2)CC1 13963,c1(C(=O)NC2CCC2NC(=O)C(O)c2ccsc2)ccc2c(c1)CCCS2(=O)=O 13964,C1(CNC(c2csc(C)c2C)=O)CN(C(=O)CCC#N)CCC1C 13965,C1(C(N(CCN(C(C)C)C(c2ccc(CCO)cc2)=O)C)=O)C2CC2C2CC12 13966,C1(CNC(c2ccn(CCOC)n2)=O)COC(C)(C)CN1C(c1cnsc1)=O 13967,c12nc(nn1CC1CCSC1)C2.c1nc(C2CCCCC2)n(C2CCSCC2)n1 13968,C(=O)(C1=C(C(C)=O)N(CCF)C(=O)NC1c1cc(Cl)c(F)cc1F)OCC 13969,N1(C(Cc2c(C)ccs2)=O)CCC(C)(NC(=O)Cc2nnn(C(C)(C)C)n2)C1 13970,c1(C(N2CCCC(NC(c3ccc(CO)nc3)=O)CC2)=O)cn2ccnc2cn1 13971,c1(C(=O)NC(C2C(C(N3CCC(C)(N(C)CC)C3)=O)C2)C)ccc2cc[nH]c2c1 13972,C#Cc1ccc(CCCC(=O)NC2CCN(C(c3c[nH]c(=N)o3)=O)CC2C)cc1 13973,CC#CCCCC(=O)NCC1CCCCC1NC(c1oc(Br)cc1C)=O 13974,c1(C(N(CCOC)C)=O)occc1CNC(c1nccn1C(C)C)=O 13975,C(=O)(C(CN(C)C)N(C)C)NCCN(CCOC)Cc1cn(C(C)(C)C)nn1 13976,C(=O)(C1CCCc2nn[nH]c21)NCC(C)CNC(c1ncn2c1CCCC2)=O 13977,c1(C(=O)NCC2CCC(NC(C(c3cnn(C)c3)OC)=O)C2)ccc(O)nc1Cl 13978,Cn1c(C(=O)NCC(C2CCOC2)NC(c2cnc3n2CCS3)=O)cccc1=O 13979,CCCCC(C)CCC(=O)N1CCC(F)C(NC(c2ncoc2C2CC2)=O)C1 13980,c1(C(=O)NCC(c2ccccc2)N(C)C(c2cnn(C)c2)=O)n[nH]c2c1CCC2 13981,C1(CNC(C=Cc2n(CC)ncc2)=O)CCN(C(=O)C(C)(C)SC)CC1C 13982,Cc1cc(C(N2CCCC2CNC(C2(c3cccnc3Cl)CC2)=O)=O)cc(F)c1C 13983,C(=O)(C(F)(CNC(=O)CC1CC(CC)=NO1)C(C)C)N1C(CC(C)=O)CCCC1 13984,CC(C)C(CNC(=O)CC1(O)CCC1)C(=O)NCC1C2CCCCCC12 13985,c1(C(C)C(=O)NCCNC(=O)Cc2csc(NC=O)n2)ccc(OC(F)F)cc1 13986,c1(OCC(N2CCC(N3CCCC3=O)CC2)=O)ccc(Br)cc1OCC(F)(F)F 13987,C1(C(=O)NC2CCN(C(c3cnc(CC(C)(C)C)s3)=O)C2)CCC2(CC1)CC2 13988,Cc1cnc(C)c(C(N2CC(N(C(=O)C(C3CCOCC3)C)C)C(C)(C)C2)=O)c1 13989,N1(C(C(COC)OC)=O)CCCC(NC(C2(O)CC2)=O)CCC1 13990,CC1(NC(=O)CC23CCC2CN(C(=O)C2=CCCCO2)C3)CCC(O)CC1 13991,CCCC(O)C(=O)NC(C(=O)N1CCC(C(C)(C)C)CC1)C(C)C 13992,c1(C(=O)OC)[nH]c(=NCC(C)CNC(=O)C(O)C(C)c2ccccc2F)sc1C 13993,CCCCCCC(C)C(=O)NC1CC(C(=O)NCc2nnn(C)n2)=CC1O 13994,Cc1c[nH]nc1CC(=O)N(CCCN(C)C(C1CN(C2CCOCC2)C1)=O)C 13995,N1(C(c2c(C)nn(CC)c2C)=O)CC2CCCC2(NC(=O)Cn2cncc2C)C1 13996,CC1(C)C(c2ccc(Br)cc2)CCN1C(C1CCN(C(=O)C(C)(C)C)CC1)=O 13997,c1(C(=O)NC2(C(=O)NCC(C)Cn3cccn3)CC2C)cc([N+](=O)[O-])n[nH]1 13998,C1(c2cn(CC(=O)N(CC)CC)nn2)CSCCN1C(=O)C(N1CCC(C)CC1)=O 13999,N1(C(C(C(CC)O)C)=O)CCOC2(CCN(C(C3(C)CCCN(C)C3)=O)C2)C1 14000,c1(C(=O)NCCCN(C(C(C)n2cccn2)=O)C)ccc(S(=O)(=O)CF)nc1 14001,c1(C(=O)NC2C(O)CCN(C(CCCCC#C)=O)C2)cc(Cl)cc(Cl)c1O 14002,n1(CC)nc(C(C)C)cc1C(C)C.c12ccc(nc1)C(=O)N1CC2(O)C1 14003,c1(C(=O)NCC2(O)CCCN(Cc3nc(CC)sc3)C2)c(F)cc(Cl)cc1F 14004,C1(C(N(C)CC2CCN(C)C2)=O)CC2(CCC2)CN1C(c1ccc(C#N)s1)=O 14005,CCC(C)CCC(=O)NCc1nc(C)c(C(=O)NCC2(CC)CCCC2)o1 14006,C(=O)(C1=NOC2(CCN(c3nccc(Br)n3)C2)C1)Nc1cc(C)c(C)c(C)c1 14007,C1(C(=O)NCC(C(C)C)NC(c2csc(C(F)F)n2)=O)CC(=O)N(C)C1 14008,c1(C(=O)OC)ccc2sccc2c1.N12CCOC(C1)C2C(C)C 14009,N1(C(c2ccc(CC)s2)=O)CCC(F)CC1C(N1CCN(C)CC1C1CC1)=O 14010,C(CC1=CCCCC1)N(C)C(C1CN(C(c2nnn(C)c2N)=O)CCO1)=O 14011,C(=O)(C(C)(C)CF)N(C1CCN(C(C2CCNC2=O)=O)CC1)C 14012,c1(C(N2CC(C(C)NC(CSc3n(C)nnn3)=O)C2)=O)ccc(N)cc1O 14013,c1(C(N2CC(CNC(CC3(OC)CC3)=O)C(O)C2)=O)cc(C)c(Cl)cc1F 14014,Cn1c(CN(CCO)Cc2ccc(C(N)=O)cc2)nnc1-c1cnc(O)nc1 14015,c1(NC2CN(C(C)=O)C2)[nH]c(=NC(C)c2cnc[nH]2)nc2sccc12 14016,N1(C(=O)Cn2cnnc2)CC2CC(N=c3ccnc(CO)[nH]3)CC1C2 14017,C(=O)(CC(C)(C(F)F)N(C)C)N(C(C)CNC(c1cocc1Br)=O)C 14018,N1(C(CC(CC)c2ccc(C)cc2)=O)CCC2(CC1)CN(C(=O)CCC(C)=O)C2 14019,C(c1ccc(Cl)cc1Cl)=CC(=O)N(C1CCCN(C(C)=O)C1)C 14020,C(=O)(C(CCC1CCC1)NC(=O)C1=CCCC1)NC(c1ccc(O)cn1)C 14021,C1(C2(NC(C34CC(CN3C(=O)CC(C)F)C4)=O)CC2)(OC)CCC1 14022,C1(C(N2CC(O)(CNC(C(CC)NC(N)=O)=O)C2)=O)CC2(CCC2O)C1 14023,C12(C(N(C3CCN(C(C(C)OCC)=O)C3)C)=O)CCC(OC)(CC1)CC2 14024,S(=O)(=O)(CCC(=O)NCC1COCCN1C(c1ncnn1C(C)C)=O)NC 14025,N1(C(CCOCC#C)=O)CCC(NC(c2ccc3nc[nH]c3c2)=O)C2(CCC2)C1 14026,C=Cc1ccc(C(N2CCCC(CNC(=O)CC3CC(CC)=NO3)CC2)=O)cc1 14027,c1(C(=O)NCCC2CCC(NC(c3ccc(Cl)o3)=O)C2)cccc2cc[nH]c12 14028,Cc1c(Cl)cc(CN2CCCC(C(=O)NC3CC(O)C3)CC2)cc1I 14029,c1(C(N2CCN(C(c3nc(CC)oc3)=O)CC2CC)=O)c(C)cc(Br)cc1C 14030,c1(CC)cc(C(=O)NC2CC(C(=O)NC3C=CCC3)C2)ccn1 14031,c1(C(=O)NCC23CC(NC(CN(CCC)C)=O)(C2)C3)ccc2cccnc2c1 14032,C1(CC=C)(NC(=O)CC2CCC(C3CC3)O2)CCN(C(=O)CC(C)(F)F)CC1 14033,N1(C(c2c[nH]c(=NC)s2)=O)CCCC12CCCN(C(=O)CC1CC(C)(C)C1)C2 14034,c1(C(=O)NCC(CNC(C2C(OC)CC2)=O)(C)C)cccc(SC)c1[N+](=O)[O-] 14035,C(CCCCN(C(=O)CC(C)n1cc(Br)cn1)C)NC(C=C(C)C1CC1)=O 14036,n1(CCC)cc(Cl)c(C(=O)NC(C)CN(C(c2cccc(F)c2)=O)CC)n1 14037,c1(OC)cc(C)c(C(=O)NCC2CCC3(CN(C(=O)CC(C)SC)C3)O2)c(C)c1 14038,C1(NC(C(CC=C)NC(=O)C=CCOC)=O)CC(C)(C)OC1(C)C 14039,C1(N(C(c2cc(CC)on2)=O)C)CCCC(N(C(=O)CCCN2CCCC2)C)C1 14040,CCC(N)C(C)(C)C(=O)NC1(CO)CCN(Cc2cccc(C(F)(F)F)c2)CC1 14041,N1(C(CC(C(C)OC)NC(c2c(CC)oc(C)c2)=O)=O)CC=C(C(C)(C)C)CC1 14042,C(c1ccc(OCC)c(Cl)c1)=CC(N1CC(NC(COCC)=O)C(C)C1)=O 14043,C12(NC(CC3(CSC)CC3)=O)CC3CC(C1)CC(NC(C1CCC(C)O1)=O)(C3)C2 14044,C1(C(N(CC(=C)C)CC(=C)C)=O)CCCC(NC(c2ccc(C3CC3)nc2)=O)C1 14045,N1(C(c2n(C)ncc2Cl)=O)CC(O)CCC1C(=O)NCC1(CC2CCC2)CC1 14046,c1(OC)ccccc1CC1CCCN1C(=O)C(C)NC(=O)CCc1ccc(C)cn1 14047,N1(C(C(CC=CC)C)=O)C(C(N2CCCC2C(O)CC)=O)CCC12CC2 14048,C1(C(=O)NCC2(SC)CCC2)CC(F)CN(C(=O)C(c2cccn2C)=O)C1 14049,Cc1cccc(C(=O)NCCC23CCC2CN(C(c2nocc2Br)=O)C3)c1O 14050,c1(CNC(C2COCCN2CC)=O)coc2cc(N)c(-c3ccc(CO)s3)cc12 14051,CC1=C(C(=O)N2CCC(NC(=O)CC(O)CC(C)C)C(O)C2)C(=O)OC1(C)C 14052,c1(C(=O)NC2CC(NC(=O)COCCOCCO)C2)ccc(F)c(O)c1F 14053,C(=O)(CCN=c1cc(NCC2CC(C3CC3)C2)nc[nH]1)N(C)C 14054,c1(SCC(=O)NCC2(F)CC(NC(C3C4CC4C4CC34)=O)C2)cccc[n+]1[O-] 14055,N1(C(C(C=CC)O)=O)CCC2CC12C(=O)N(C(C)CC1CC1)C 14056,N1(C(=O)CSc2n[nH]c(O)n2)CCN2CCNCC2C1 14057,C1(CNC(C(C=CCCC)O)=O)(CO)CCN(C(=O)CSCCN(C)C)C1 14058,N1(CC(=O)NC(CNC(CC=C)=O)C(C)C)C(=O)NC(C)(COC)C1=O 14059,c1(CC2C(C(=O)NCc3cnc(C)[nH]3)COC2)ccc(Br)cc1 14060,c1(C(N2C(C(C)NC(=O)C(O)C3CCC3)CCC2)=O)cc2c[nH]cnc-2n1 14061,c1(OC)ccc(S(=O)(=O)N2CCCC(C)(C(=O)Nc3c[nH]nc3C#N)C2)cc1Br 14062,C(=O)(CCCC(F)(F)F)NCCCN1CCC(NC(C(NOC)=O)=O)C1 14063,C1(NC(CNC(=O)OC)=O)(CNC(c2cnc[nH]2)=O)CCCCCC1 14064,c1(OC)ccc(CN2CCCC(C(=O)N(C)CC3CCCCC3)CC2)c(Cl)n1 14065,C(CN=C(NCC(=O)N(C)C)NCC1CCOC1)(c1ccc(F)cc1)OC 14066,CCCC(C)(CC)C(=O)NC1CC(CCNC(=O)C(C)(CC)CC)C1 14067,C1(NC(C(CC)N(CC)CC)=O)C2CN(C(c3cccnn3)=O)CC12 14068,N1(C(C(CCCC)=O)=O)CCOC2(CCN(C(=O)C=Cc3cccs3)C2)C1 14069,CC1(NC(C2Cc3nccn3C2)=O)CCN(C(c2cc(Cl)cs2)=O)CC1 14070,Cc1cc(CC(=O)NCCN(C(C23CCCCC2C3)=O)CC2CC2)n(C)n1 14071,CCCCC(O)C(C)C(=O)N1CCN(C(=O)CC2CCSC2)CC1C(C)(C)C 14072,c1(C(=O)NC2C(NC(C3CN(C)C(=O)N3)=O)CCC2)cccc(C(N)=O)c1F 14073,c1(OC(F)F)ccc2c(c1)CN(C1CC(=C3CCC3)C1)C2 14074,c1(C(N(C(C)CNC(=O)Cn2cnnc2O)CC)=O)ccc(N2CC=CC2)cc1 14075,c1(C(c2n(CCOCC)nnn2)NCCC2CC=CC2)cc(C)nn1C 14076,c1(C(=O)NC2CC(C)(NC(C3N(C)C(=O)CC3)=O)C2)ccc2nc(O)[nH]c2n1 14077,N1(C(CSCC=C)=O)CC(NC(c2cnoc2-c2ccc(Cl)s2)=O)CC1(C)CC 14078,Cc1c(C(=O)NCC2(C)CCCN2C(=O)C2=COCCC2)nn2c1OCCC2 14079,C1(C(c2ccccc2)NC(=O)C(=O)NCC(=C2CCSCC2)F)CCCC(=O)N1 14080,c1(OC)c(F)ccc(-c2ccc(CC(=O)NC(C)C#N)cc2F)c1F 14081,c1(-c2nc(C(C)OCC)nn2-c2nc(C)nn2C)onc2cc(C)ccc12 14082,c1(NC(c2n(CCCC(=O)OCC)nnn2)(C)CC)ccc2c(c1)CCCS2 14083,c1(C(N(C2CC(NC(=O)CC3CCC3)C2)C)=O)ccc(OCC(F)(F)F)c(Cl)c1 14084,c1(C(=O)NC2CC3CN(C(C4(CCOC)CCC4)=O)CC32)ccc(S(C)=O)cc1 14085,C1(NC(CCCCOC)=O)C2CC3C1C3C2C(=O)NCCN1CCOCC1C 14086,Cc1nn(C(C)(C)C)c(C)c1C(=O)NC1CCCCN(Cc2cncnc2)C1 14087,c1(C(N2C(CNC(C(C)n3ccnn3)=O)CC2)=O)cccc(Nc2nccs2)c1 14088,C(C(C(=O)NC(CNC(C)=O)C1CCC1)C(F)(F)F)OC 14089,c1(N(C)C)ncc(C(=O)NC(CC(N)=O)c2cn(CC3CCCO3)nn2)cn1 14090,C(c1cccc(O)c1)=CC(=O)NCC(C)(F)CNC(C1CCCN1C1CC1)=O 14091,N1(C(=O)NCC2CCC(C)C2)c2ccc(F)cc2CCC1C 14092,CCCCC(C(=O)NC1CC2(C1)CN(C(c1cc(CC)[nH]n1)=O)C2)NC(N)=O 14093,C(=O)(CCCCCCC=C)NC(CC#C)C(=O)NCCCc1cccs1 14094,C1(NC(c2ccc(C#C)o2)=O)(CO)CCCN(C(=O)CCCc2ccccn2)C1 14095,c1(C(=O)NC2CCCN(C(CC(COC)C)=O)C2C)ccc2c(c1)C(=O)NC2=O 14096,c1(C(N2CC(NC(C3C(C)C3c3ccccc3)=O)C2)=O)nccnc1Cl 14097,C1(CNC(C2(C)CCCS2)=O)CCC(F)(CNC(=O)CN2CCCCC2)C1 14098,N1(C(C(CC=C)OC)=O)CCCC(O)(CCNC(C2(O)CCCCCC2)=O)C1 14099,C(=O)(C(C)(C)C(N)=O)NCCCC(C)NC(=O)C(C)c1ccco1 14100,C1(CC)(NC(c2ccc(Cl)c(OC)c2)=O)CCCN(C(=O)CCc2cn[nH]c2)C1 14101,CC1CN(C(=O)CC(C)(C)O)CC2(CCN(C(c3ccc(=O)n(C)n3)=O)C2)O1 14102,c1(CCC)cccc(C(=O)N(CCCNC(C2C3CN(C)CC23)=O)C)c1 14103,c1(C(=O)NC(C2CCCN2C(=O)CN=S(C)(C)=O)(C)C)ncc2c(F)cccn12 14104,CC(C)C(C(=O)NCCNC(c1cccnc1-c1ccc(F)cc1)=O)C1CCC1 14105,C1(CNC(c2c(CC)c[nH]c2)=O)C(C)CCN1C(c1n[nH]c(C)c1C)=O 14106,C12(NC(CCCC3C(C)C3)=O)CCC(C(=O)NC34CC=CC(C3)OC4)(CC1)C2 14107,C1(NC(c2c(CC)noc2)=O)CN(C(c2cccc(N)n2)=O)CC(C)(C)C1 14108,C1(C2(O)CN(C(c3cccc(OC)c3)=O)C2)(CNC(C(COCC)C)=O)CC1 14109,C(=O)(CCCCCCNC(=O)C(=Cc1cn[nH]c1)C)N1C(CCOC)CCCC1 14110,CCCCC(C)(F)C(=O)N1CC2(CCN(C(c3cocc3Br)=O)C2)C1 14111,c1(SCC)ccccc1-c1ccc(N2CCN(C(c3ncnn3C)=O)CC2)nc1 14112,C1(C(C)C)CN(C(c2ccc(Cl)nc2)=O)CCN1C(c1cn(C(C)C)nn1)=O 14113,c1(C(=O)NCCC(CNC(c2ccc(CO)s2)=O)OC)cccc(C)n1 14114,N1(C(C2C3CN(C(C(C)O)=O)CC2CC3)=O)CCc2ccc(Cl)cc2C(C)C1 14115,C1(CNC(C2C(CC)C2)=O)CN(C(c2cc(C(=O)C(C)C)c[nH]2)=O)CCC1(F)F 14116,C12(C(=O)NCCCCNC(c3cn(C)nc3Cl)=O)CCC(CC1)C(C)(C)O2 14117,c1(SC)ccc(C=CC(N2CC(CNC(C3CC4CC4C3)=O)C(C)C2)=O)o1 14118,CC1CCCCCCN1C(=O)C(C)N(C(=O)CCN1CCOC1=O)C1CC1 14119,Cc1c(NCCn2cnc(Br)n2)nc[nH]c1=NCCc1sccc1Br 14120,N1(C(c2c(C)nns2)=O)CCC(N2CCN(C(c3cccnc3Cl)=O)CC2)CC1 14121,C(CC(O)C(F)(F)F)NC(C1N(C(Cc2ccn(C)c2)=O)CCC1)=O 14122,c1(C(N2CCC(N)(CC(=O)OC)C2)=O)cc(Br)c(O)nc1C 14123,N1(C(c2cnc(C(C)C)nc2)=O)CC(C)CCC1CNC(c1ccc(F)o1)=O 14124,c1(NC(C(CC)NC(=O)C2CC2)=O)ccc(CNC(=O)CC23CCCC2C3)cn1 14125,N1(C(c2n[nH]c(C)c2N)=O)CCCCC(NC(=O)C=Cc2ccc(C(F)F)o2)C1 14126,c1(CNC(Cn2c(C)cc(C(F)F)n2)=O)n[nH]c2c1CN(C(=O)C=CCO)CC2 14127,c1(COC)ccc(C(=O)N(C(C)CNC(C2(c3cccnc3)CCC2)=O)C)s1 14128,N1(C(C(C(C)O)(F)F)=O)CC2(C1)CN(C(=O)CC(=O)NC1CC1)CCO2 14129,c1(C(C(=O)NCC(C)N(C)C(c2cnccn2)=O)(C)F)ccccc1F 14130,CS(=O)CCC(O)C(=O)NC1CC(CNC(c2cncc(F)c2Cl)=O)C1 14131,C1(C2(O)CN(C(C3CCCC(C(N)=O)C3)=O)C2)(CNC(C(C)(C)CO)=O)CC1 14132,C(=O)(C(C)(C)C(O)C(C)C)NCC1(F)CCN(C(c2n(CC=C)ccc2)=O)C1 14133,CC1CN(C(=O)C=CC2CCCC2)CC(C)N1C(C1CCC(C2CC2)C1)=O 14134,c1(NC(Cc2cccc(C)n2)C)ncnc(NCC2C=CCN2S(C)(=O)=O)c1C 14135,CCCCC(C(=O)NCC1C(C)(C)C1(F)F)NC(c1cc(C2CC2)[nH]n1)=O 14136,Cc1nn(C)cc1C(=O)NC(Cc1cnc[nH]1)C(=O)NCC1CC(C2CC2)C1 14137,C(=O)(C(CC(=C)C)NC(c1c[nH]nc1OC)=O)NCCCCCC=C 14138,C1CN(C=O)CCO1.n1(C2(N(C)CC)CC2)cc(C(O)C2CC2)nn1 14139,C1(O)(C(C)NC(c2cnc(C3CC3)s2)=O)CCN(C(c2cnc(S)nc2)=O)C1 14140,C=CCC(CC)C(=O)N(C1CN(C(c2ccnn2C)=O)CC1(C)C)C 14141,C1(C(c2occ(C(N3CCC(NC(C)=O)C3)=O)c2)=O)CCN(C(=O)C(C)C)CC1 14142,C1(C(=O)OC)CC12CCC(NC(=O)Nc1ccc(F)cc1Cl)CC2 14143,CC(C)(C)C#CC(=O)NCC1CN(C(=O)C=Cc2ccsc2)CC1(F)F 14144,N1(C(C(CN(C(Cc2cc(C)sc2)=O)C)C)=O)CCC2(COC(=O)N2)C1 14145,N1(C(C(C)NC=O)=O)CC(O)(CCNC(=O)Cc2ccsc2)C1 14146,C1(N(C(CCC=C)=O)CCO)CCCN(C(C2(C)CC=CC2)=O)C1 14147,C(=O)(C(C)(CC(C)C)NC(=O)OC(C)(C)C)N1C(CNC(C(C=C)(F)F)=O)CC1 14148,C1(C)(C(N2CCC(N(C(C(CC)O)=O)CC)C2)=O)CC(C)(C)C1 14149,N1(C(C(C=CC)O)=O)CCC(CC(=O)NCCCOC(=N)O)CC1 14150,N1(C(c2cc(C)ns2)=O)CCC2CC2(C(=O)NCc2ncccc2F)CC1 14151,Cc1nsc(-c2nnc(CC(C(CCN(C)C)N(C)C)c3ccccc3)o2)n1 14152,N1(CC(=O)Nc2c(OC)cccc2)CCCC(=O)C1C 14153,c1(OC)cc(NC(C2CC(NC(C3CC(OC)C3)=O)C2)=O)cc(F)c1 14154,c1(C(=O)NC(CC)CNC(C2CCN2C2CCCC2)=O)ccc2ncccc2c1 14155,c1(OCC)cc(C(=O)NC(C)CN(C(=O)Cc2c[nH]ccc2=O)CC)ccn1 14156,c1(C(=O)NCC(N(C)C(C2(C(F)(F)F)CCCC2)=O)C2CC2)ccnc(OC)c1 14157,N1(C(C(C)OCCC=C)=O)CCC(N(C)C(c2ccn(CC(C)C)n2)=O)C1 14158,c1(C(=O)NCCCN(C(=O)CCNC=O)CC)cnn[nH]1.C(C(N)=O)S 14159,N1(C(COCC(=O)OC)=O)CC2CC(NC(=O)C(C)Cn3cccn3)C1C2 14160,C1(S(=O)(=O)NN2CCCC2)(C(C2CCCN2CC(F)F)=O)CCC1 14161,N1(C(C(=O)Nc2cc(C)c(-n3cncn3)cc2)=O)CC2CC(NC(N)=O)CC1C2 14162,C#Cc1ccc(NCc2ccnc(CO)c2)cc1C#N 14163,CC(C)C(O)C(=O)N1CC2CC1(CNC(=O)CC1CC3(CC3)C1)C2 14164,c1(-c2ccc(-c3n(-c4ccn(CC=C)n4)ccn3)s2)cccc(S(C)(=O)=O)c1 14165,C1(NC(c2c(OC)oc(C)n2)=O)CN(C(=O)CC2CCC(=O)NC2)CC1C1CC1 14166,C1(NC(=O)Nc2cnc(O)c(C(F)(F)F)c2)CN(c2ncns2)CC2(CCC2)C1 14167,c1(NC(C)=O)ncc(S(=O)(=O)Nc2cc(Br)ncc2F)s1.C12CCN(C1)C2=O 14168,c1(OCC(CN2C(CNC(c3c(COC)ncs3)=O)CCC2)O)cccc(C)c1 14169,N1(CCNC(C2(C)CCCS2)=O)CCCN(C(C2(n3cccn3)CCC2)=O)CC1 14170,CC1CCCC(C)N(C(C2(CO)CCN(C(=O)CCn3ccnc3)C2)=O)C1 14171,CC(O)C(C(=O)N(C1CC1)CC1CCN(C(c2ncoc2C(C)C)=O)CC1)N(C)C 14172,C1(CC(=O)NC2CCCC(CNC(c3cccc[n+]3[O-])=O)C2)CCS(=O)(=O)CC1 14173,N1(Cc2cccc(C(=O)NC(C)CCC(F)F)n2)C(=O)c2ccccc2C1=O 14174,N1(C(C2(C)C(C)(C)C2)=O)CCC(CC(=O)NCC2CC3C=CC2O3)CC1 14175,N#CC1(C(=O)NC2CCCC(C(=O)NCc3ccncn3)C2)CC12CCC2 14176,Cc1cccnc1C(C)NC(c1ccc(-n2cc(-c3ccn(C)n3)nn2)nc1)=O 14177,c1(C(N2CC(CCC=C)(C(N3CCCCCCC3)=O)C2)=O)ccc2[nH]ccc2n1 14178,Cc1ccc2c(NC(C3CCN3Cc3cnc4ccc(F)cn34)=O)cccc2n1 14179,C1(C(=O)NCCCc2onc(C)n2)CN(C(=O)CCCNC(=O)C2CC2)CCO1 14180,N1(C(CC(C=C)C)=O)CCC(CNC(c2cccc(C(=O)OC)n2)=O)C1(C)C 14181,c1(CC)cc(CC(N2CCCC2C(C)NC(c2cn(C(C)(C)C)cn2)=O)=O)on1 14182,n1(CC(=O)NCC(CNC(CC)=O)F)cnc(-c2ccccc2)n1 14183,N1(C(CN(C2CC2)CC)=O)CCC(CNC(c2ccc(O)cc2F)=O)C(CC)C1 14184,Cn1cc(C#N)cc1C(=O)NCC(O)CNC(c1coc(-c2cccnc2)n1)=O 14185,CCCC(CCCNC(C12CC(NC(c3cc(CC)cc(C)c3)=O)(C1)C2)=O)OC 14186,C1(NC(c2cc(CC)on2)=O)CC12CCN(C(=O)CNC(N)=O)CC2 14187,C(=O)(C1=CCSC1)N1C(C(C)(C)CNC(C2C(C)(C)C2(C)C)=O)CCC1 14188,C=CCC(F)(F)C(=O)NCC(C1(O)CCN(C(c2coc(C(N)=O)c2)=O)C1)C 14189,CC(CCNC(C1CN(C(c2ccoc2)=O)C(C)(C)C1)=O)CC(C)(C)C 14190,CCCN(Cc1ccc(O)cc1)N1Cc2ccc(C(C)=O)cc2C1 14191,N1(C(C(C)Cn2ccnc2)=O)CC(NC(=O)CCN(C)CCO)CC2(CC2)C1 14192,N1(C(CC(c2ccc(OC)cc2)C)=O)C2CCC(C(=O)O)C1CC2 14193,CCCC(C)(O)C(=O)N1CC(C(C)NC(c2ccc(=O)n(O)c2)=O)C1 14194,c1(C(N2CC(CCCCNC(C=COCC)=O)C2)=O)cc(C)c(C)nc1C 14195,C1(NC(COCC=C)=O)CC1C1CCN(C(C2CCc3nn[nH]c3C2)=O)CC1 14196,N1(C(CSCC=C)=O)CC2CCCN(C(=O)C(C)Oc3cccc(C)c3)C2C1 14197,c1(CC(=O)N(C)CC2CCCN(C(=O)C=CCO)C2)coc2ccccc12 14198,N1(C(CCC(=O)OC)=O)CCN(C(c2ccc(C)cc2Cl)=O)C(C(F)F)C1 14199,N1(C(C(C2(O)CCC2)NC(c2ccc(C#N)[nH]2)=O)=O)CCC2(COC(=O)N2)C1 14200,C1(O)(CC)CCN(C(c2cc(C(N)=O)co2)C(=O)NC(C)CC)C1 14201,c1(CN2CC3(CCC(C(N4CC(F)(F)C4)=O)O3)C2)c(F)ccc(Br)c1F 14202,c1(NC(C23CCCCC2C3)=O)ccc(NC(c2nccs2)=O)c(F)c1 14203,c1(C(=O)NCC(=C2CN(C(CC3CCC(OC)C3)=O)C2)F)cc(C)ncc1C 14204,N1(C(c2cnc(C(C)C)[nH]2)=O)CC2C(CNC(=O)CCCc3ccccc3)C2C1 14205,c1(C(=O)NCC(C)(C)F)cc(-c2cncc(F)c2)nc2ccccc12 14206,c1(C(N2CC(NC(CC3CC(OC)C3(C)C)=O)(CO)C2)=O)ccc(Cl)c(N)c1 14207,N1(C(C)=O)C=Cc2ccccc2C1CC(=O)NC1CC(n2cc(C(=O)O)nn2)C1 14208,c1(CC)ccc(C(=O)NC(C)CNC(=O)CS(=O)(=O)C2CC2)cc1[N+](=O)[O-] 14209,C1(C2CN(C(c3sccc3F)=O)C2)(NC(c2ccc(O)nc2Cl)=O)CC1 14210,CCCC(O)(CCC)CC(=O)NC(C)CN(C)C(C1CCn2nccc2C1)=O 14211,N1(C(C(C)=C(C)C)=O)C2CCC1C(F)C(NC(C1(N(C)C)CCN(C)CC1)=O)C2 14212,CC1=NOC2(C1)CC(C(N1CC(NC(c3cc(C)on3)=O)CC(C)C1)=O)C2 14213,C(CNC(C1(O)CCCC1)=O)(CC(C)C)NC(Cc1cnc(C)s1)=O 14214,C1(F)(C(=O)OC)CN(C(c2ccco2)=O)CC1c1cccnc1 14215,c1(C(=O)NCC(Cn2cc(COC(C)C(=O)O)nn2)OC)cccc(F)c1C 14216,c1(OC)cc(NC(=O)CC2(C)CC2(Cl)Cl)ncn1.C12CCC(CC1)CN(CC)C2=O 14217,C1(C(=O)NCCCNC(COCCCC)=O)CCCCC1F 14218,Cc1ccc2sc(C(N3CCC(CO)(NC(=O)C(=O)C(C)(C)C)CC3)=O)cc2c1 14219,C1(NC(C(C)(C)CO)=O)CN(C(c2n[nH]c3ccccc23)=O)C2(CCCCC2)C1 14220,N1(C(c2ccc(CSC)cc2)=O)CC2CC(C)N(C(C3CCC3CF)=O)C2C1 14221,N1(C(c2ccc(OC)c(Br)c2)=O)CCC2(CCN(Cc3ccc(O)c(O)c3)C2)C1 14222,O=C(C#CC1CC1)NCC(C1CCCCC1)NC(c1cccc(NC(N)=O)c1)=O 14223,C1(C(CC)C)CCN(C(=O)C(C2(O)CCC2)NC(c2cccs2)=O)CC1 14224,C(=O)(C#CC1CC1)N1CCC(CC2CCN(C(CCNC(=O)OCC)=O)C2)C1 14225,c1(CC)nc(C(C)C)ccc1C(=O)NCC(CC(C)C)NC(=O)COCC1CC1 14226,C(=O)(C(C(C)NC(C1CCC(C)=C(C)C1)=O)C(C)C)N1CC=C(C)CC1 14227,C(C(C)(C)CN(C)C(c1cc(C)ns1)=O)NC(C(C1CCCC1)NC(C)=O)=O 14228,C#CCCCCCCNC(C1CC(C)CN(C(c2c[nH][nH]c2=N)=O)C1)=O 14229,Cc1cc(C(=O)NCCC2CC(NC3CC34CCOCC4)C2)ccc1[N+](=O)[O-] 14230,CON1CCC(C(=O)NC2CCCC(C(=O)NC3CC(F)(F)C3(C)C)C2)CC1 14231,c1(OC)ccc(C(=O)NCC2CC2NC(C2(CN(C)C)CCOCC2)=O)cc1 14232,N1(C(C(CC2CC2)OC)=O)CCCN(C(=O)CN2CCCCCC2)C(C)C1 14233,c12nocc1C(=O)N2.C1(CC=C)(C(=O)NCCC2(c3ccon3)CC2)CCC1 14234,C#CCCCCCC(=O)NCC(CC=C)NC(c1cc(C)nn1CC)=O 14235,N1(C(c2cc(C(C)C)[nH]n2)C(=O)NCCC(=O)OCC)CC2CC=CC1C2 14236,CC(C)CC(O)C(=O)NCC1CCCN1C(=O)C1=CCCCC1 14237,C1(C)(NC(=O)OC(C)(C)C)CN(C(=O)NC(CC)(c2nn[nH]n2)SC)C1 14238,c1(OC)cccc(CCC(=O)NC2CCCCN(C(=O)C(C)(C)C)C2)c1F 14239,c1(CC(C)NC(=O)N(CCN2CCCC2=O)CC2CC2)nccn1C 14240,C1(C(=O)NC2C(NC(COCCOCC)=O)COCC2)CC2CCCC2C1 14241,N1(c2ncnc(OC)c2C)CCOC2CN(C(c3nc(Cl)sc3Cl)=O)CC12 14242,CC1CC=CCC1C(N1CC(NC(c2ccccc2C(C)(F)F)=O)C(F)C1)=O 14243,c1(OC)ccc(CNC(=O)N(C2COCC2(C)C)C)cn1 14244,c1(CC)cc(OC)ccc1N.c12ccc(cc1)N(CC)C(=O)C2N 14245,N1(C(C2CC(OC)C2)=O)CCC2C(NC(=O)CC3CN(C)CC3O)CC12 14246,c1(OC)cscc1C(N1CCC(CCNC(C2CC2F)=O)C1)=O 14247,C1(C(=O)NCC2(C(C)NC(C3CC=CC3)=O)CC2)C=CCCC1 14248,c1(C(C)C)conc1CC(=O)NC(CNC(=O)C(C)CC1CC1)C(C)C 14249,c1(OC)cccc(NC(c2c(C(F)(F)F)ccc(Cl)c2Cl)=O)c1[N+](=O)[O-] 14250,C=CCCCCCCCC(=O)NC1CCCCC1CNC(c1ccnn1CC)=O 14251,C1(N(C)C(=O)OC(C)(C)C)(CN(CCCNc2nnn(C)n2)C)CCOCC1 14252,N1(C(C2(C(N)=O)CC2)=O)CC(C(=O)NCCc2ccc(O)cc2)C(F)C1 14253,c1(OC)ccc(C(=O)NC2CCN(C(c3cncn3C)=O)CC2C)cc1N 14254,N1(C(COCCOCC)=O)CCC(NC(=O)COCc2cccc(C)c2)CC1 14255,c1(C(c2noc(C(C)NS(C)(=O)=O)n2)C)cc2ccc(O)cc2[nH]1 14256,C=CCC(C)C(=O)NC1(CF)CCN(C(=O)C(C)NC(c2ccc(Cl)nc2)=O)C1 14257,C(=O)(CC(C(F)(F)F)P(C)(C)=O)NCCC1CC(NC(c2c(C)[nH][nH]c2=N)=O)C1 14258,CCCCCCCN(C)Cc1ccc(SCc2cn(C3CCOC3)nn2)cc1 14259,C#Cc1ncc(F)cc1NC(c1ccc(Cl)s1)c1nnnn1CC1CCCO1 14260,c1(NC(CC2CCN(C(c3nc(CC)oc3)=O)C2)=O)cc([N+](=O)[O-])ccc1CO 14261,c1(OC)c(Cl)ccc(C(=O)NC(C)C(C)NC(=O)CN2C(=O)CN(C)C2=O)c1F 14262,C(c1nc2ccccc2o1)=CC(=O)NCC1(F)CCN(C(C(C)OCC)=O)CC1 14263,N1(C(C(CC)c2ccccc2)=O)CC2(CC(NC(c3c(C)ncn3C)=O)CO2)C1 14264,Cc1[nH]nc(Cl)c1C(=O)NC1(C2CCCCN2C(=O)C(C)CC2CC2)CC1 14265,CC1CN(C(=O)CC2(C)CCCO2)CC1CNC(c1nn(C)cc1Cl)=O 14266,C1(Cc2cn(CCCCSC)nn2)CCCC(C)C1 14267,C(=O)(C1=NNC(=O)CC1)N(CCCNC(=O)Cc1cc(C)cc(C)c1)CC 14268,c1(CC(=O)NC2C=CCN(C(c3c(C(=O)OC)cco3)=O)C2)cc(F)ccc1Cl 14269,N1(C(C(C(C)C)n2cccc2)=O)CCC2(CCCN(C(=O)C(C)CC(N)=O)C2)C1 14270,c1(CCC(=O)NCCCN(C(=O)C(C)C2=CCCC2)CC)nc2ncccn2n1 14271,c1(N2C3(CNC(=O)C4=NOCC4)CCC2CC3)ncnc2sc3ccccc3c12 14272,N1(CC(=C)Br)CCN(C2(C(N)=O)CCCC2)CC1 14273,C(C(F)(C(=O)N(C)Cc1cccc(C)c1)C(C)C)NC(C=CCC)=O 14274,C1(CC)CC(CC(N2CC(NC(=O)C(=O)OC(C)(C)C)C2)=O)CCO1 14275,N1(C(CC2C(C(=O)OC)C2(F)F)=O)CCOC(C)(CNC(=O)C(=O)NC2CC2)C1 14276,c1(N(C(=O)CN(C(c2c[nH][nH]c2=N)=O)C2CC2)C)ccccc1O 14277,N1(C(c2c(C)nn[nH]2)=O)CCC(F)C(NC(c2cc(Br)ncc2Br)=O)C1 14278,c1(NC(c2c(N(C3CCCCC3)C)cccc2)=O)csc2ccccc12 14279,c1(C(N(C2CCN(Cc3cnn(C)c3)C2)CCC)=O)ncoc1C 14280,c1(OC(CC)=O)ccc(OCC)cc1C(N1CCCCC1CCO)=O.C1C(=O)N1 14281,N1(C(c2c(CC)nn(C)c2)=O)CCCC(F)(C(N2CCCC2(C)CO)=O)C1 14282,c1(C(=O)NC2CC(NC(C(C(C)C)N(CC)CC)=O)C(O)C2)cc(F)cnc1O 14283,C1(NC(C2CCN(C)C2)=O)C2CN(Cc3ncc(Br)s3)CC12 14284,c1(CC(N2CCC(C)(NC(C=Cc3ccc(C)o3)=O)C2)=O)cccc([N+](=O)[O-])c1 14285,c1(NC(C2CCN(C(c3ccncc3)=O)C2)C)ncc([N+](=O)[O-])c(=N)[nH]1 14286,N1(C(C)(C)C)CCCC(C(=O)NC2(c3ccc(Br)cc3)CCCO2)C1=O 14287,O=C(C1CCCc2c[nH]nc21)NC1CN(C(c2cc(F)c(F)cc2O)=O)CC1F 14288,Cc1cnc(Cl)c(C(=O)NC(C2CCN(C(c3ccco3)=O)C2)C)c1 14289,c1(C(=O)NCC2(CNC(CC(COC)C)=O)CCCCC2)cnn2ncccc12 14290,C1(OC)CCC(C(=O)NC2CCC(NC(=O)C(C)CC3CC3)C2)CC1 14291,C1(C(=O)NC2CC(CNC(c3nc(C)oc3C)=O)CC2O)CC2OC1C1CC21 14292,c1(C(N(C(C)CNC(=O)Cc2cc(C3CC3)on2)C)=O)ncc(C#N)cc1F 14293,c1(OCC(=O)N=CC(O)C(=O)OCC)cccnc1OC 14294,n1(CC=C)cc(C(=O)NC2(C(N3CC(C)(OC(C)=O)C3)=O)CCC2)cn1 14295,C1(CC(c2n(C)nnn2)N(C2CC2)CC2C(C)(C)C2(C)C)CC(F)(F)C(=O)N1 14296,N1(C(CC(CC2CC2)NC(=O)CCc2ccsc2)=O)CC2CCCC(O)C2C1 14297,C(=O)(CC(C)CC(C)C)NCC(C(=O)N(C(CC)CO)CC)C(C)C 14298,N1(C(c2ccnc(C)c2N)=O)CCCC(C)(C)C1C(=O)NCCC(C)C(F)F 14299,O(S(=O)(=O)c1cccc2c1OC(C)C2)CC(S(CC)(=O)=O)(C)C 14300,CC1(C)OC2CC(C(=O)NCC3CN(C(=O)Cc4nnc(O)s4)CC3O)CC2O1 14301,Cc1n[nH]c(C)c1CC(=O)NC1CCC(CNC(c2cnsn2)=O)C1 14302,CCCC(=O)NCC(=O)NCC(F)CNC(=O)Cn1cccn1 14303,C1(CNC(c2cccc(SC)c2)=O)CN(C(c2cnns2)=O)CCC1C(F)(F)F 14304,N1(C(C(CCCC)(C)F)=O)CCC2(CCC(NC(C3CCCC3OC)=O)C2)C1 14305,N1(C(C(C(C)C)NC(C)=O)=O)CCC2CCC(NC(=O)CC3(C)CC3)C1C2 14306,c1(C(=O)NC(CCCNC(C(C)OC)=O)C)cccc(SC)c1[N+](=O)[O-] 14307,C#Cc1cncc(C(N2CCCC2(C(=O)Nc2ccc(O)cc2CC)CC)=O)c1 14308,N1(C(c2c(C)sc(O)n2)=O)CCC2(CC1)CC(NC(c1ccc(O)nn1)=O)C2 14309,N1(C(CSc2n(C)cnn2)=O)CCC(C)(C)C(NC(=O)CSC(F)(F)F)C1 14310,C1(NC(C2CCCC2)=O)COCCN(C(=O)CC(O)Cc2ccccc2)C1 14311,C1(C(=O)NC(CC)CNC(=O)CN2CCCCC2)CCC2(CCC2)OC1 14312,c1(C(=O)NCCN(C(c2nsnc2O)=O)CC)cc(S(=O)(=O)CC)ccc1OC 14313,CC1CC(c2cn(CCN3CCNC3=O)nn2)CCN1C(C1CS(=O)(=O)C1)=O 14314,N1(C(C(C)S)=O)CCN(c2ncc(-c3ccc(CO)cc3)cn2)CC1 14315,Cc1n[nH]c(C)c1CO.C12CN(CC1C(F)F)C(=O)c1ccn(n1)CC(=O)N2C 14316,c1(C(N(C)CC2COCCN2C(=O)CC2(C)CCCC2)=O)cccc(S(C)=O)c1 14317,N(C1c2ccccc2CC1NC(=O)C(O)P(C)(C)=O)C(C(OC)OC)=O 14318,c1(OC)c(C(=O)NC2CC(C)CN(C(c3cnc(Cl)nc3)=O)C2)cccc1C#N 14319,C1(CN(C2CCCN(C(c3c(C)nc(CC)o3)=O)C2)C)CC12CCCCC2 14320,N1(C(CCC=CC(C)C)=O)CCN(C(C2CCCN2C2CCOCC2)=O)CC1C 14321,N1(C(C(C)=C2CCC2)=O)CCC2C(CCCN2C(=O)Cn2cnnn2)C1 14322,C(S(=O)CC(=O)N1CCC(C(=O)NCC(C)C)CC1)c1ccc(COC)o1 14323,C1(NC(C(CCC)C)=O)CN(C(=O)C(C)Oc2cc(C)ccc2Cl)CC(F)(F)C1 14324,Cc1c(C(=O)NC2CC(C)CN(C(C3CCC(C)CC3)=O)C2)cccc1F 14325,C1(NC(c2occ(C(=O)OC)c2)=O)C2CC(CN(C(c3csnn3)=O)C2)C1CO 14326,CCCC(C(=O)NCC(C(C)C)NC(c1cn(CC(=O)N(C)C)nn1)=O)N(C)C 14327,N1(C(CC2OCC(C)(C)OC2)=O)CC2=C(C1)CN(C(C1CC1C(=O)OC)=O)C2 14328,N1(C(c2ccc(CC)o2)=O)CCN(C(CNC(C2CC2C)=O)C(F)F)CC1 14329,Cc1ncc(C#N)cc1NC(=O)C(O)CCNC(C1C2CCCCCC12)=O 14330,N1(C(C2CCCCN(C(c3cc(COC)[nH]n3)=O)C2)=O)CCC(O)C(C)(C)C1 14331,CC1(C)CC(C(=O)NCCC2CN(CCCS(C)(=O)=O)CCS2(=O)=O)CC(C)(C)O1 14332,C1(C(N(CCCNC(=O)Cc2nn(C)cc2Br)CC)=O)CC2CC(=O)C1C2 14333,C#CCCCC(C)C(=O)N(CCNC(C1CCCSC1C)=O)CC 14334,Cc1cc(F)c(C(=O)N(CCN(C)C(C2CCCC3CC23)=O)C(C)C)cc1F 14335,C1(C#N)(C(=O)NCC(CNC(c2c(OCC)cccn2)=O)OC)CCCCC1 14336,c1(C(=O)NCC(C)NC(C2CC3CC3C2)=O)ccncc1I 14337,C1(C2CCC2)(C(=O)NC2CCC(CCNC(c3ccn(CC)c3C)=O)C2)CCC1 14338,c1(CN2CC3N(C(c4c(OC)ccc(F)c4)=O)C(C3)C2)cccc(F)c1C#N 14339,C1(CNC(CCOCCC)=O)CC(F)(F)CN1C(=O)C(c1ccn(C)n1)C 14340,c1(OC)cccc(CC(N2CC(NC(C3CC4(CC4)C3)=O)C(SC)C2)=O)c1F 14341,N1(C(C(C)=C(C)C)=O)CC2CC3CC2C1C3NC(=O)Cc1ccoc1 14342,Cc1ccccc1COC1CC1NC(=O)Cn1cnnn1.N12CCC(C1)C2=O 14343,C1(N(CCCC)C(c2ccc(CO)o2)=O)CCN(C(=O)CNS(=O)(=O)NC)CC1 14344,C1(CNC(C(COC)O)=O)CC2(CO1)CN(C(=O)CSSC)C2 14345,c1(-c2cn(CCC(N3CCN(C4CCSC4)CC3)C)nn2)cc(C)nc(C)c1 14346,c1(C(=O)NCC(C)N(C(=O)Cc2cn(C)nn2)C)ccc2ncnn2n1 14347,Cc1nnc2n1CC(C(=O)NC(CNC(c1nccn3cnnc13)=O)C(C)C)C2 14348,C1(C(N(C2CN(C(Cc3c(C)noc3)=O)CC23CC3)C)=O)CC(=O)N(C)C(=O)N1 14349,C#Cc1cccc(C(=O)Nc2nc(CNC(=O)Nc3ccc(F)c(Cl)c3)cs2)c1 14350,c1(C(N(CC(C)N(C(=O)C2=CCSC2)C)C)=O)cc2c([N+](=O)[O-])cccc2[nH]1 14351,C1(CC)(NC(C2OCCO2)=O)CCCN(C(=O)CC2CCCCC(=O)N2)C1 14352,C1(NC(c2ncc(OC)cn2)=O)CC(N=c2[nH]nc(C3CC3)s2)C12CCC2 14353,C12(CNC(C34OC(C)(C)C(C3)C4)=O)CN(C(=O)CCn3cncn3)CC1CCO2 14354,O(S(=O)(=O)c1ccc(C#N)cc1)c1ccc(F)cc1F.C(=O)(CON)N(C(C)=O)CC 14355,C(=O)(C1=CC2(CCN(C(=O)CC3COC(=O)C3)C2)C1)NC(CC#C)CC#C 14356,C1(C(N2CC(COC)(CNC(=O)Cc3cnoc3)C2)=O)CCC(C)(C)O1 14357,C12(CNC(c3c(C)nsc3)=O)CCCC1CN(C(=O)CCc1ccccc1)C2 14358,c1(CNC(N2CCC(C)C2)=O)nc2cc(Cl)c(Cl)cc2[nH]1 14359,O=C(CCCC1(c2ccccc2)CC1)N(C1CCCCC1)CCO 14360,C(c1cccc(Cl)c1)=CC(=O)NC(c1sc(C(=O)OCC)c(C)n1)C 14361,c1(C(N2CCCC(CNC(C(CC)NC(C)=O)=O)C2)=O)csc2ncnc(O)c12 14362,c1(C(=O)NCC2CC(O)(CNC(=O)C(F)CC3CC3)C2)cc(F)cc(Cl)c1 14363,CCCC(C(=O)NCCN(c1ncnc(=N)[nH]1)CC)S(N)(=O)=O 14364,c1(C(=O)NC2CC3CC(NC(c4c(C)cns4)=O)C2C3)nc2ccccc2[nH]1 14365,c1(C(=O)Nc2c(OC)ccc(O)c2)coc2c1CN(C(C1CCC(F)C1)=O)C2 14366,C1(C)(C(N2CC(SCc3ccc(CC)s3)C(O)C2)=O)Cc2ccccc2C1 14367,C1(NC(CCCC(C)=O)=O)CCN(C)C12CCCN(C(C1CCC(=O)N1)=O)C2 14368,Cc1cc(C(N2CCC(NC(=O)C(F)(F)C(F)(F)F)CC2C)=O)ncc1C#N 14369,CCC(O)C(F)(F)C(=O)N1CCN(C(=O)CN2CCNC(=O)C2)C(CC(F)F)C1 14370,C1(NC(c2c(OC)c(F)ncc2)=O)CC2(CCN(C(c3sc(C)nc3C)=O)C2)C1 14371,N1(C(C(C)O)=O)C2CCC1CN(C(C1CCN(CC(F)(F)F)CC1)=O)CC2 14372,N1(C(c2cc(N)cc(OC)c2C(=O)OC)=O)CC2CCCC(NC(=O)C(C)Br)C2C1 14373,C(C(=O)NC1C=CC(C(=O)NCCc2c[nH]nc2O)C1)(C(C)C)OCC 14374,C1(NC(CC(C(=C)C)OCC)=O)C2CCCN(C(C3CCCC3F)=O)C2C1(C)C 14375,c1(OC)ccc(Br)c(CN2CCCC(C(=O)NCC3CN(C)CCO3)CC2)n1 14376,Cn1nnc2cc(C(N3CCC(C4CCCN4c4ccnc(Cl)n4)C3)=O)cnc12 14377,Cc1cc(N)n2ncc(C(N3CCC3CNC(C3(C(=O)N(C)C)CC3)=O)=O)c2n1 14378,CC(C)CC(C)(O)C(=O)NCC1CCCCN1C(=O)Cc1ccc(Br)nc1 14379,c1(C(N2C3C(NC(c4cnc(COC)s4)=O)CC(C3)C2)=O)cc(F)cc(N)c1F 14380,C1(NC(c2cc(C)no2)=O)CC(Nc2nccc(CO)n2)C1(C)C 14381,O=C(C(O)C(F)(F)F)N1CCOCCC1C(=O)NOCCCC(F)(F)F 14382,CCC(C#N)C(=O)NC(C(=O)NCc1ncc(C)s1)C1CCC1 14383,c1(C(=O)NCC(CC)(C)N2CCOCC2)cc(S(N)(=O)=O)c(Cl)o1 14384,c1(-c2nc(CC3ON=C(C)C3)sc2)c(F)cccc1Cl.N12CCCC(C1)C2=O 14385,C=C(CNC(c1nnnn1CCSC)(C)COCC(F)(F)F)C1CCOCC1 14386,C1(N(C(c2cnc(O)o2)=O)CC)CCCN(C(c2cnccc2C(F)F)=O)CC1 14387,c1(NC(=O)NCCc2ccc(C)o2)cccc(N=c2cc[nH]cc2)c1 14388,N1(C(c2c(C)cc(SC)o2)=O)CC2CC(NC(C3CCCC3(C)C)=O)C2C1 14389,C1(CNC(c2cc(C(N)=O)[nH]n2)=O)CCN(C(=O)C(O)C2CC2)CCC1(F)F 14390,C1(NC(CNS(CCCC)(=O)=O)=O)CCN(C(=O)CCCC)CC1O 14391,N1(C(CC(C)N(C(C(CCCC)O)=O)C)=O)CC2(CCCCCC2)C1 14392,O=C(C(O)c1ccsc1)NC1(C(=O)NCC(Cl)=CCl)CC1 14393,C1(C(=O)NCCC2N(C(CCN(CCC)C)=O)CCOC2)CCC(C)=C(C)C1 14394,N1(C(c2n(C(C)C)ncc2)=O)CCCC2(CCC(NC(c3cccnc3)=O)C2)C1 14395,C(=O)(C1=NOC2(CCC2)C1)N(CCCC(=O)NCCOCC(C)(C)O)C 14396,CC1=CCC(N=c2ccc(Br)c(S(=O)(=O)NC3CCC4(C3)CC4(F)F)[nH]2)CC1 14397,C(c1cc(Cl)c2c(c1)OCO2)=CC(=O)NCC(CO)NC(C1(C)CC1(F)F)=O 14398,S(=O)(=O)(c1ccc(Cl)cc1)N(C(CCC)C)C(c1cnn(C2CC2)c1)=O 14399,c1(OC)cc(C(N2CC(C(=O)N(C3CCC(O)CC3)C)C(C)C2)=O)nn1C 14400,c1(C(=O)NCC2C3CN(C(C(C(C)C)OC)=O)C2C3)cc(Cl)cc2cccnc12 14401,C12(NC(C3CCCO3)=O)CC(CNC(=O)C(O)C3CCC3)(C1)OC21CCOCC1 14402,C(=O)(CC(C(F)(F)F)NC(=O)CCn1ccc(C)n1)NCCC1ON=C(C)C1 14403,Cn1ncc2cccc(C(N3CCC4CN(C(c5ccnc(O)c5)=O)CC34)=O)c12 14404,CC1(C#CC(=O)NCCc2ocnc2CNC(=O)CC2CCC3CC23)COC1 14405,S(=O)(=O)(c1cc(C(F)(F)F)cc(C(F)(F)F)c1)N1CC(c2cc(N)on2)OCC1 14406,c1(C(N2CC=CC(NC(c3cc(SC)ncc3)=O)C2)=O)oc2ccccc2c1Cl 14407,c1(CC)cccc(F)c1C(=O)NCCOCCCNC(C1C(F)(F)C12CC2)=O 14408,C#CCCCCC(=O)NC(Cn1cccn1)C(=O)NC1CCC1(C)C 14409,c1(C(=O)NC(CNC(C(CSC)C)=O)(C)C2CC2)cnc(O)c(C(F)(F)F)c1 14410,Cc1cc(=O)n(CCC(N2CCC(NC(c3cnns3)=O)C2C(C)(C)C)=O)cn1 14411,C=CCC(CO)NC(=O)CC1(NC(C2CCC(=O)C2)=O)CC1 14412,C1(CN(C)C(C23CSCC2C3)=O)CCN(C(C2CC23CCC3)=O)CC1 14413,C1(C(C)CNC(=O)C(=O)NCC2CC2)CCCN(C(=O)C=CC2CC2)C1 14414,C1(CNC(CCCC#C)=O)COC(C)(C)CN1C(C1CCC(F)(F)C1)=O 14415,C=CC(CCC)CC(=O)NCCC1CCCN(C(C2(C(C)C)CCC2)=O)C1 14416,c1(C(=O)NCCNC(c2c(C)c3c(s2)ccs3)=O)cc2c(s1)CC(C)CC2C 14417,c1(N2C(CCNC(c3c(C)cc(C)o3)=O)CCC2)nc2ccccc2s1 14418,n1(CCCC)c(CC(=O)NCC2(C)CN(C(=O)C(CO)OC)C2)nc2ccccc12 14419,c1(CC)nn(C)cc1CNC(=O)CC1CCN1C(=O)C(C)NC(=O)OC 14420,c1(C(N2CC(NC(CCSCC)=O)C(C)CC2)=O)nn2c(c1C)OCCC2 14421,CCC(CC)(CC)C(=O)N1CCC(N(C)C(c2csc(C3CCCC3)n2)=O)C1 14422,C#Cc1ccc(C(=O)N(C2CCCN(C(c3ccn(C4CCC4)n3)=O)C2)C)nc1 14423,C(CNC(c1cccn(C)c1=O)=O)(CC(F)(F)F)NC(C(=Cc1cccs1)C)=O 14424,c1(CNC(=O)C#CC2CCC2)nc2c(s1)CN(C(=O)C=Cc1ccc(Cl)s1)CC2 14425,c1(OC)ccc(S(=O)(=O)NCC2CCC(CSC)CC2)cc1 14426,C(CCCC(=O)OC(C1(C)CC1)=O)(C(=O)OC)N1CCCC(OCCC)C1 14427,N(C1CCCn2ncnc21)C(C1C2CN(C(=O)C3=C(Cl)CCCC3)CC21)=O 14428,CN1N=CC(CC(=O)NC2CC(CCC(N3CCOCC3CO)=O)C2)C1=O 14429,CC1=C(C(=O)NC2(C)CN(C(C3C(C)(C)C3(F)F)=O)C2)CCCO1 14430,c1(-c2n(CC)ncc2)nc(C(N2CCCN(CC3CC3)CC2)=O)ccc1F 14431,N1(C(CCC(=C)C)=O)CCC(NC(c2ccc(OC(F)F)cn2)=O)CC1C1CC1 14432,C(c1ccc(Br)cc1)=CC(=O)NC(C)CCCNC(=O)CP(C)(C)=O 14433,N1(C(COCc2cc(C)no2)=O)CCCC1(C)CNC(c1nccs1)=O 14434,c1(SC)nc(N2CCC(NC(c3cccnc3O)=O)CC2)c(Br)c(C)n1 14435,C(=O)(C(O)(C(C)C)C(F)(F)F)NCC1(CNC(c2cc(OC)ns2)=O)CC1 14436,CC1CC(NC(c2cccc(Br)c2)=O)CCN1C(=O)CC1CCCCN1C 14437,C#CC1CCC(C(=O)NCCN(C(=O)C(C)N2CC(C)C2)CCOC)CC1 14438,C12(C(N3C4C(CNC(=O)CSc5ccc(O)cc5)C(C4)C3)=O)CCCC1OCC2 14439,C1(O)(CC)CCN(C(C2C=CC(NC(c3n[nH]cc3C)=O)C2)=O)CC1 14440,C(CC(C(=O)NC1CC(n2ccnn2)C1)NC(C1CC(CF)C1)=O)OC 14441,C1(C(=O)NC2C(CCC)C2)CCCN(C(c2ccccc2OCC)=O)CCC1 14442,Cn1[nH]nnc1=NCCCCCCNC(C1(c2cccc(F)c2)CC1)=O 14443,c1(C(N2CC(C(N3CCC(c4ccco4)C3)=O)(CC)C2)=O)ccc(C)nc1 14444,c1(CCC)ncc(C(C(=O)NC(C)C)C(C(=O)N(CC(C2CC2)NC)C)=O)s1 14445,N1(C(c2ccc(Cl)cc2)C(=O)NCCC#N)CCCN2CCCCC12 14446,c1(C(=O)NC2(CN(C(=O)CC3CCCO3)C)CC2)ncccc1OCC(F)(F)F 14447,Cc1nn(CCO)cc1C(=O)NCC1CCCC1NC(c1cc(O)nn1C)=O 14448,c1(CC)cc(C)c(-c2nc(COC(C)(C)C)nn2Cc2ccncc2)o1 14449,C(=O)(C(C)(CC)CC)NCc1ccc(C(N(CC=C)CC)=O)o1 14450,Cc1ccc(NC(C23CC(NC(=O)CCN4CCCC4)(C2)C3)=O)c(C(F)(F)F)c1 14451,N1(C(=O)NCc2cc(C)nn2C)CCN(C(C2CC2CC(C)C)=O)CC1 14452,C1(C)(CNC(COCCOCC)=O)CCCN1c1ncncc1Br 14453,c1(C(N2CCC(C(C)NC(C(CC#C)C)=O)CC2)=O)cc(C)ccc1N 14454,c1(OC)cc(C(=O)NC2CC(NC(c3c(C)nn(C)c3N)=O)C2)nc(C)c1 14455,N1(C(C2(NC(C34CSCC3C4)=O)C(C)CCC2)=O)CCCCC(CO)C1 14456,O=S(=O)(c1ccc2nc(N3CCC(O)C(F)C3)ccc2c1)N1C2CCC1CC2 14457,c1(CC(=O)NC(C2CCN(C(c3cncnc3)=O)CC2)C)ccccc1S(C)=O 14458,C1(n2c(-c3nnn(Cc4cccs4)c3CC)nc(CCC)n2)C(C)CCCC1C 14459,N1(C(c2c(OC)nc(C)nc2)=O)CCCN(C(c2ccc(F)cc2C)=O)CC1C 14460,c1(NC(CCC)C)cc(=NCCc2cnc3ncccn23)[nH]c(COC)n1 14461,CCCC(CCC)CC(=O)N1CCOCC1CNC(=O)C(C)(CC)CO 14462,CONC(=O)CNC(=O)CCC1CC(NC(c2coc(C(N)=O)c2)=O)C1 14463,C1(SC(C)C)(OC)CC(=O)N(CCC)C1CCC(C)C 14464,C1(NC(c2cc(C3CC3)cs2)=O)CCN(C(C2CCCCS2(=O)=O)=O)CC(O)C1 14465,N1(C(CCOCC#C)=O)CCN(C(=O)CCCc2cccnc2)C2CC12 14466,C1(N(C(=O)OCC)C)CCN(N2CCN(CCC(C)(C)C)C(=O)C2)CC1 14467,CC(CC#N)N=c1cc[nH]cc1S(=O)(=O)NCC1(OC(F)F)CCCCCC1 14468,N1(C(C=CCNC(C2CCC3CC3CC2)=O)=O)C(CO)CCC12CCC2 14469,c1(C(=O)NC2CCC(CCNC(C3(CCCC)CC3)=O)C2)cc(C)c(O)c(C)c1 14470,c1(SCC(C)=CC(=O)OCCC(=O)N(C)C)cccnc1C(F)(F)F 14471,c1(C(=O)NCC2C(C)(C)CCN2C(=O)CSCCC#N)cnn2c1OCC(O)C2 14472,C(=O)(C(C)CC(C)C)N1CCC(N(C(C(C(=O)OCC)F)=O)C)CC1 14473,c1(CNC23CC(C(=O)NCCNCCO)(C2)C3)cc(Br)cc(F)c1F 14474,N1(C(C(C)n2cncn2)=O)CC2C(N(C(=O)CCCN(C)C)C)C2C1 14475,c1(CC(=O)NCC2C3CN(C(c4n(CC)ccc4)=O)CC32)nsc2ccccc12 14476,N(C(=S)N1CCC1c1ccnn1C)c1scc(C)n1.C12=CC=C(C=C1)C2 14477,Cn1cc(CC(=O)NCC2(C)CCCN2C(=O)CCC2CCC2)c(Cl)n1 14478,CCC(C)(COC)CNC(=O)CONC(=O)C=Cc1cncs1 14479,C(C)(C)(CC(=O)NC(C)CC(C)NC(=O)CCCCc1cnc[nH]1)OC 14480,C1(C(N2CC(N(C(C(CC)(C)O)=O)C)C2)=O)CC(c2cccnc2)=NO1 14481,C1(NC(=O)C(O)c2ccsc2)CN(C(c2cc(C3CCC3)no2)=O)CC1O 14482,c1(OC)cc(F)c(C(N2CC(CNC(c3cnn4ccn(C)c34)=O)C2)=O)cc1N 14483,C1(CC)C(C(=O)NCc2cccc(OC)c2)CCN1C(c1cnn(C)c1Cl)=O 14484,N1(C(C(F)(F)C2(OC)CCC2)=O)CCC(NC(=O)C2=CCCCC2)CC(C)(C)C1 14485,N1(C(C(C)OC2CCCCC2)=O)CCC(C)C(NC(=O)C(C)(C)CO)C1 14486,CCC(CC)C(=O)N(C)CC1CN(C(c2ncn(C(C)(C)C)n2)=O)CCO1 14487,c1(C(=O)OCC)cnn2c1CN(C(C1CC1NC(=O)CN(C)C)=O)CC2 14488,N1(C(CC(=C)C)=O)CCC2CCN(C(C3CC(C)(C)CN3C)=O)CC12 14489,c1(SCCC(=O)N(C2CCN(C(c3coc(C(F)(F)F)n3)=O)C2)C)ccccn1 14490,C#Cc1cccc(C(=O)NC2CCN(C(C3COC3)=O)C(C3CC3)C2)c1Cl 14491,c1(N(CC(C)C(C)(C)C)C)nc2c(c(=NC3COC(C)(C)C3)[nH]1)COCC2 14492,C(C(CO)(CO)NC(c1cncnc1)=O)N(C(C1C(OC)C1)=O)C 14493,c1(C(=O)Nc2ccc(OCC(=O)NCC)cc2)c(C#N)cnn1C 14494,C1(NC(C(CC(=O)OC)C)=O)CC2CCC1CC2NC(=O)CC1(CS(C)(=O)=O)CC1 14495,c1(C(=O)NC23C(CN(C(CC4C(C)(C)CC4)=O)C2)C3)cccc2c1OCCO2 14496,C1(C(N2CC(CNC(c3cc(OC)no3)=O)(COC)C2)=O)CCCCN1C(C)C 14497,C(CC(C)(C)C(=O)N1CCCC(CN(C(=O)Cc2csc(Cl)c2)C)C1)OC 14498,C1(C(=O)NCCCC(C)O)CCCCCC1NC(C1CCC(F)CC1)=O 14499,N1(C(COCc2cc(C)no2)=O)CCCC(C(=O)NCC2(C)CC=CCO2)C1 14500,N1(C(c2c(C)coc2)=O)CCCN(C(=O)C(CO)N(C)C)CC1c1ccccc1 14501,N=c1cc[nH]cc1C(=O)NC1CC1NC(c1ccn(CC(F)(F)F)n1)=O 14502,C1(O)(CNC(Cc2cncc(C)c2)=O)CCCN(C(c2nn(C)c(C)c2Cl)=O)C1 14503,c1(CC(=O)NCCN2CCN(C(CSCCCC)=O)CC2)c(C)nc(O)nc1C 14504,Cc1nc(CNC(C2CC2c2ccco2)C)sc1C(=O)O 14505,Cc1c[nH]cc1C(=O)N(C)CCOCCNC(C1CC1CF)=O 14506,C12(CNC(C=CC)=O)CC(NC(=O)CC(CC)SC)(C1)C(C)(C)O2 14507,C1(N)(CC)CCCN(C(=O)C(N2CCCC(C(=O)Sc3cccnc3)C2)=O)C1 14508,CCCC(CC)CCC(=O)NC12CC(C(N3CC(O)(CO)C3)=O)(C1)C2 14509,CCCCS(=O)(=O)NCC(=O)NC1CC1CNC(c1ccc(C(F)(F)F)cn1)=O 14510,C(=O)(C(CC(N)=O)NC(c1cc(C)n(C)c1)=O)NCCCOCCCC 14511,c1(C(CC)C)nc(-c2coc(C)n2)n(C(C)C(C)(C)C)n1 14512,N1(C(CSCC=C)=O)CCCN(C(C2(C3CC3)CC2)=O)CC1c1ccccc1 14513,N1(C(C2CCC(C)O2)=O)CC=CC(NC(=O)C(=O)N(C)C)C1 14514,N1(C(CC2N(C(C)C)CCC2)=O)CCOC2(C1)CN(C(c1cnn(C)c1F)=O)C2 14515,C1(NC(c2c(C(C)O)cccc2)=O)CCN(C(C2CC(O)C2)=O)C(C)C1 14516,C1(C2(O)CCOCC2)(C(=O)NC2(C)CN(C(=O)Cc3cccc(N)c3N)C2)CC1 14517,CCC(C)(C)CCCC(=O)NC1CCN(C(c2cc(C)cc(F)c2)=O)C12CC2 14518,c1(C(=O)NCCC2CC(NC(=O)C(F)(F)c3nccs3)C2)ccc(CO)c(Cl)c1 14519,C1(C(=O)NC2(CF)CCN(C(c3nc(CC)sc3)=O)C2)CCCC1S(C)(=O)=O 14520,c1(C(N(C(=O)CC2CC=CCC2)C(C)C)=O)cncc2nc[nH]c12 14521,C=Cc1ccccc1NC(=O)CC(=C)C 14522,Cc1c(C(=O)NC2CC2NC(=O)CCC2CCCC2)cc(-c2ccccc2)n1C 14523,N1(C(CC2(OC)CCC2)=O)CCN(C(c2cccc(F)c2O)=O)C2(CC2)C1 14524,N1(CC(=O)NC)CCC2CCN(Cc3nc(-c4ccccc4)n[nH]3)CC12 14525,C1(O)(C(C)NC(COCCNC(c2c(C)scc2)=O)=O)CCCCC1 14526,C1(C(=O)NCCN(C(=O)CO)CCC)CCC(C(F)(F)F)O1 14527,CC1CN(C(C2CC3CCC2C3)=O)CCC1CNC(c1cnn(C(F)(F)F)c1)=O 14528,c1(CC(N2CC3(CC(CNC(C(C)(O)C4CC4)=O)C3)C2)=O)csc2ccccc12 14529,Cc1cc(-c2cc(C(=O)NC(c3ccccc3Cl)CO)ccn2)cc(O)c1 14530,N1(C(C(C2CC2)SC)=O)CC2(C(=O)N(CC3=CCSC3)C)CC1CO2 14531,N(C1CC2(CN(C(=O)C=C3CC3)C2)n2ccnc21)C(C1C(=O)NCC1)=O 14532,C1(C(N(CCOCCN(C)Cc2nc(CC)oc2)C)=O)CCc2nnc(O)n2C1 14533,Cc1cccc(OCC(=O)NCCC(C)NC(=O)CCCC#N)c1 14534,CCCCC(C(=O)N1CCN(C(c2cc(C(C)(C)C)oc2C)=O)CC1CC)N(C)C 14535,c1(C(C(C)C)Nc2c(O)ccc(C#C)c2)ccc2ccccc2c1 14536,C(=O)(C(C)S(N)(=O)=O)N1CC(O)(CNC(c2c(C)n(-c3cnn(C)c3)nn2)=O)C1 14537,C(=O)(CC1C(=O)Nc2ccccc21)NCC1N(C(CC(C)(C)CC(F)F)=O)CC1 14538,C1(C2CCNCC2)(C(=O)NCC(Cc2ccccc2C(F)(F)F)CO)CCC1 14539,C(=O)(C(C)CC(C)(F)F)N(C(CCNC(CC(C=C)(C)C)=O)C)C 14540,C1(NC(C(=O)NC(c2cccnc2Br)C)=O)CCCN2CCCCC12 14541,C(=O)(CCCCC(N)=O)N1CCC(CNC(CN2CCCC(N(C)C)C2)=O)CC1 14542,CC1OC2(C(=O)NC3CC(O)(CNC(=O)CN(C)C)C3)CCC1CC2 14543,c1(C(C)(C)C)nc(N2CC=CC(NC(c3ccccc3CO)=O)C2)[nH]c(=N)n1 14544,CCC(C)(C)C(C)CC(=O)NC1CC2CCC1(NC(=O)CN(CC(C)(C)C)C)C2 14545,c1(SC)cscc1C(N1CCC(NC(C2CC(SC)C2)=O)C1)=O 14546,c1(C(C(F)(F)F)C(=O)OC(c2ccc(C)o2)C(N2CC(F)(F)C2)=O)ccc(O)cc1 14547,C1(NC(C(CCC)C)=O)CC2(CCN(c3cc(Cl)nc(SC)n3)CC2)C1 14548,C1(C(N)=O)CCC(CCC(=O)NCC2CCN2C(c2ccsc2Cl)=O)O1 14549,c1(OC)ccncc1CC(=O)NC1COCC1NC(c1csc(C(F)F)n1)=O 14550,c1(C(N2CC3(CCN3C(c3cc(Cl)sc3Cl)=O)C2)=O)cc2n(c1)CCOC2 14551,N1(C(CC=CCC)=O)CCCC(OC(N2CCC2C)=O)C1 14552,c1(CC(=O)N(CC(C)N(C(CC(C=C)CC)=O)C)C)coc2c(Cl)c(Cl)ccc12 14553,C1(NC(CSCc2c(C)nc[nH]2)=O)CC2CN(C(=O)CO)CC2C1 14554,c1(CNC(c2c(C)n[nH]c2)=O)ccc(CNC(c2c[nH]c(C(F)(F)F)c2)=O)cc1 14555,C1(C(=O)NCc2c(CNC(c3n[nH]c(C)c3O)=O)cccc2)CC12CCCCC2 14556,C(=O)(C(CCC=C)NC(c1nnccc1C)=O)NCCCCC#C 14557,C1(CNC(=O)C=Cc2cn[nH]c2)(NC(C2SCCCS2)=O)CC2CCC1C2 14558,c1(CCCC)ccc(C(=O)OCC(=O)CCc2ccccc2)cc1[N+](=O)[O-] 14559,O=C(CS(=O)(=O)CCO)NC(C1CCCC1)CNC(c1ccn2ccccc12)=O 14560,CCC(CC)N(CCC(=O)NC(C1CN(C(=O)Cc2cn[nH]c2)C1)C)C 14561,c1(C(N(C2CCN(C(CSCC#C)=O)C2)C)=O)cc(C)nc(N2CCCC2)n1 14562,C1(NC(c2c(C)ncs2)=O)CCCOC12CCN(C(=O)CC1CC=CCC1)CC2 14563,N1(C(CCCCC#N)=O)CCN(C(=O)Cc2noc3ccccc23)CC(CO)C1 14564,C1(OC(c2cn(Cc3ccoc3C(=O)O)nn2)C)C=CCCC1C(=O)N(C)C 14565,CC1CN(C(N2CCC(CC(=O)OC(C)(C)C)C2)=O)CC1C(=O)Nc1nc[nH]n1 14566,C1(CNC(C(COC)(F)F)=O)CN(C(=O)C(C)NC(C)=O)C2(CCC2)C1 14567,C(=O)(C(C)(C)CC(C)C)N1CCN(C2C(NC(C=NOC)=O)CCC2)CC1 14568,N1(C(COC)=O)CCCC1CCNC(C1C(C)C1C)=O 14569,C(=O)(C(C)(C)C(F)F)NC1CC2(C(NC(c3cc(COC)cn3C)=O)C2)C1 14570,c1(N(C(C)=O)C)cccc(NC(=O)CC(c2cn(C)nc2C(F)(F)F)C)c1 14571,C1(NC(C2CC(N(C)CC)C2)=O)CCCC(NC(c2cncc(F)c2)=O)CC1 14572,C12(C(N3CCC(CNC(C4(CC5CC5)CC4)=O)C3)=O)CCCCC1OCC2 14573,C1(C(=O)NC2(CO)CCC(C)(C)C2)CN(C(C2CCO2)=O)CC1C1CC1 14574,c1(C(=O)NCC2N(C(C(C)(C)OC(C)=O)=O)CCC2)cccn2nccc12 14575,CSC1=C(C(=O)NCC2(C)CCCN2C(=O)Cc2ccc(C)cc2C)CCCC1 14576,Cc1c(C(=O)NC2CN(C(C3(c4ccsc4)CC3)=O)C2)cccc1[N+](=O)[O-] 14577,c1(C(N(C)CCNC(c2ccc(N)c(Cl)c2)=O)=O)nsc2ccccc12 14578,c1(C(=O)NCCCCCNC(CC(=O)OC)=O)cccc(C)n1 14579,O=C(CCC(CF)CF)N1CCC(NC(C2(c3ccno3)CC2)=O)C(OC)C1.C1CC1 14580,C(CCN(C)C(=O)N(C1CCC1(C)C)C)(C(C)(C)C)OC(C)=O.OCC 14581,N1(C(c2ccc(C)n2C)=O)CCCC2C1CCCN2C(=O)C(F)F 14582,c1(C(=O)NC2COCCN(C(C(CC(=O)OC)C)=O)C2)cnn2ccncc12 14583,c1(C(N2CC(CNC(CSCCOC)=O)C2)=O)nc(N(C)C)nc(=N)[nH]1 14584,C1(NC(CC(=O)OC)=O)CC(O)CN(C(=O)CCNC(C2CCC2)=O)C1 14585,Cc1ccc(C)c(C(N2CCN(C)C(C(N3CCC(OC4CC4)CC3)=O)C2)=O)n1 14586,c1(CCCC=C)ccc(C(=O)N(C)CC2(O)CN(C(=O)CC3CC34CC4)C2)cc1 14587,c1(OCC(N2CCC(NC(=O)C=CSc3nc[nH]n3)C2)=O)cccc(Cl)c1 14588,CCCN=C(NCCN1CC(C)CC(C)C1)N1CCC(COC)C1 14589,c1(C(=O)NC2CN(C(c3c(SC)cc(C)cc3)=O)C(C)C2)cc(C)n(C)c(=O)c1 14590,C1(C)(CC)CC(C(N2CC(N(C(=O)CCc3cc[nH]n3)C)C2)=O)C1 14591,c1(C(=O)NCCN(C(C2CC(OC)C2)=O)C)cccc(C#CC2CC2)c1 14592,C12(O)CCCN(C1)C(=O)NC2.N1(C(C)C(=O)NCC2CC2F)CCCCCC1 14593,c1(C(=O)NCC(C)(C)CNC(C2CC(=O)NC(=O)C2)=O)ccc2cccnc2n1 14594,CCCCN=C(NCCNS(C)(=O)=O)N1CCCC(CN(S(C)(=O)=O)C)C1 14595,C1(C(=O)NCC(C#C)CC)(CNC(C2CCCN2C(C)=O)=O)CC2(CC2)C1 14596,N1(C(C(C)(C)C(N)=O)=O)CC2CCC(CNC(=O)CCCCCC#N)(C2)C1 14597,C(=O)(C1SCCc2sccc21)N1CC(C(C)NC(C23CC4CC2C3C4O)=O)C1 14598,N1(C(CCCOCC)=O)CCN(C(C2(CN(C)C)CCCC2)=O)CC1C1CC1 14599,c1(C(=O)NC2CN(C(C3CCCCO3)=O)C2)cc([N+](=O)[O-])c2nsnc2c1 14600,c1(NC(NC(C)C)=S)ccc(Br)nc1Br.C1(O)CCCCO1 14601,CC(C)CCCCCC(=O)N1CC2(c3cn(C(C)C)nn3)CC1C2.C(=O)C(O)C(C)CC 14602,c1(C(N2CC(C)C(CNC(=O)CNS(N)(=O)=O)CC2)=O)c[nH]c2cc(O)ccc12 14603,Cc1cc(Br)cnc1C(N1CCCC1CC1CC1)C(=O)NCCC#N 14604,C(=O)(C(C)C(=O)NCc1ccc(C(=O)NC2CC(=O)N(O)C2)nc1)OC 14605,c1(CCC)ccc(C=CC(=O)N(CCC(C(C)C)NC(=O)C(O)CCC)C)cc1 14606,Cc1ccc(F)c(CNC(C2CCC(NC(c3cnc(Cl)c(Cl)c3)=O)C2)=O)c1F 14607,C(=O)(C(F)C(F)(F)F)NCCC1N(C(c2cc(C(C)(C)O)ncc2)=O)CCCC1 14608,CCC(CC)(CCNC(c1c(C)noc1N)=O)NC(c1cc(C)c(CC)s1)=O 14609,N1(C(COC)=O)CC(C)(C)CCC1CNC(=O)CS(=O)(=O)CC1CCCO1 14610,Cc1cnccc1C(C(=O)NCC(C)C)N(CC(N1CCCCC1)C)C 14611,N1(C(c2nc(C)oc2)=O)CC(NC(c2cc(C)c(Br)o2)=O)CCC(O)C1 14612,c1(OCCCC(=O)N(C2CCCN(C(C(CC)(C)F)=O)C2)C)ccc(F)cc1F 14613,N1(C(=O)NC(CCCC)CO)C(C(N2CCN(CCC)CC2)=O)C2CC(F)C1C2 14614,C1(NC(C(C)n2cccn2)=O)CCC(NC(=O)C=Cc2cccs2)C1 14615,n1(CCOC)nc(C(N2CCN(C(C3OCC3(C)C)=O)CC2CF)=O)ccc1=O 14616,N1(C(c2cncc(OC)n2)=O)CCCN(C(=O)C2=CCC2)CC1c1ccccc1 14617,N1(C(C(N2CCNC2=O)C)=O)CC2(CC(NC(c3cncnc3)=O)c3nccn32)C1 14618,C(=O)(CCC(F)(F)F)N1CC(NC(CN2CC(C)(C)C2)=O)C(CC2CC2)C1 14619,C1(CC(=O)NCC2C(C(=O)NCC3(C(C)(F)F)CC3)COC2)CCCCCC1 14620,CC1CCC2(CN1C(=O)NCCCn1ccccc1=O)OCc1ccccc12 14621,C=CCCN=C(NCCC(=O)N(C)C)NCC1CC(OC(F)(F)F)C1 14622,C1(N(C)C(c2coc(C(F)F)n2)=O)CCN(C(c2cc(Br)n(C)c2)=O)CC1 14623,N1(C(c2sccc2CO)=O)CCN(C(=O)C=CC2CC2)CC1 14624,CC(C)(C(=O)NCC=CCNC(c1csc(O)n1)=O)C1CCCC1 14625,C(=O)(C(CC(F)F)NC(=O)C(C)NC=O)N(CCO)CC 14626,c12c[nH]c3cc(ccc13)NC(=O)C(=O)NCCC2.C1(C(=O)OC)CCC(C)(C)C1 14627,c1(C(=O)NCCN(C(c2ccc(C(C)C)o2)=O)CC)n[nH]cc1I 14628,C=C1CC(C(F)(F)F)(C(=O)NCC2CC2CNC(=O)CN)C1.C(C)(C)(C)C(=O)OC 14629,n1(CCCC)nc(C)c(C=CC(N2CCCC2CN=c2[nH]nc(C3CC3)s2)=O)c1C 14630,c1(CN2CCC(O)C(O)C2)ccc2nn[nH]c2c1 14631,C=C(C)C1CCC(C)(O)C(NCCc2ccc3c(c2)CCO3)C1 14632,N(C(=NCC(C)C)NC1CC1)Cc1ccc(OC)cc1OC(F)F 14633,C1(NC(C2C(N)CCC2)=O)CCCC(F)(F)C1 14634,c1(C(=O)NCC2CCN(C(CSC)=O)CC2C)sc2ccccc2c1Br 14635,CC(C)CC(C)(C(N)=O)NC(c1ccc(CNC(C2CCC(=O)N2C)=O)nc1)=O 14636,Cc1cc(=O)oc(C)c1C(=O)NCCC(C)NC(=O)CCC=CC(C)C 14637,C1(NC(C(CCCC)NC(N)=O)=O)CCC2CCN(C(c3cc(C)co3)=O)C1C2 14638,c1(COC)cc(C(N2CC3C(NC(c4sccc4OC(F)F)=O)C3C2)=O)c(C)o1 14639,CC1CCC(C(c2nnnn2C)NC2(C)CC2)C1 14640,C1(O)(CCNC(c2c(C)nsc2N)=O)CCN(C(=O)C2=NOC(C)C2)CC1 14641,Cc1ccnc(N2CCCC(CNC(c3ccc(F)cc3C)=O)C2)c1[N+](=O)[O-] 14642,Cc1cnc2n1CCN(C(=O)C(C)(C1CC1)N(C(=O)CCc1cn(C)nn1)C)C2 14643,C(=O)C1=CC2CCCC12.N1(S(CC2(C)COC2)(=O)=O)CC2(CO)CC1(CO)C2 14644,c1(OC)ccc(CN2CCN(CCC3CCC(=O)N3)CC2)cc1 14645,C(c1cncc(O)c1)=CC(=O)NCC(CNC(c1cc(OC)ncn1)=O)O 14646,CCC(CC(=O)NCCC(C)(C)OC)N(C)C(C1CCCC(CF)C1)=O 14647,CC(C)C(F)(F)CC(=O)NC(C)(CNC(c1ccc2n[nH]cc2c1)=O)C1CCC1 14648,CC1(C)C(C(=O)NOCC2CCOC2)C1CNC(=O)CCc1nc(O)n[nH]1 14649,Cn1nccc1C(O)C(=O)NCCC1CCCN1C(=O)CSC(F)(F)F 14650,CC1CC2(CC(NC(C3CC(C)N3C(c3ccc(O)c(F)c3)=O)=O)C2)C1 14651,C=C1CCN(C(C2CC3(CC3)CO2)=O)C(C(=O)NCc2cn(C(C)C)nn2)C1 14652,N1(C(c2cnc(CC)s2)=O)CCCC(C2(NC(c3csc(C)n3)=O)CC2)C1 14653,c1(COCCOCC)cc(Cl)cnc1CC.C1(C)C(=O)N(C2CC2)CC(=O)N1 14654,c1(C(c2nnnn2-c2ccccc2)(C)NCc2cc(Br)co2)ccc[n+]([O-])c1 14655,N1(C(C(CC)n2cncn2)=O)CC(NC(=O)CC2CCN(C(C)C)CC2)C(O)C1 14656,C(=O)(C(C)C(=O)NCC(O)C(=O)N1CCC(CC2CC2)C1)OC 14657,C1(C)C(=O)N1.C1(CCOCC)(NC(CC2(N(CCC)CCOC)CC2)=O)CC1 14658,c1(CC(=O)NC2CC(NC(=O)Cc3cnn(C(F)F)c3)C2)ccc([N+](=O)[O-])cc1 14659,C1(C(N2CC3C(CN(C(Cc4cc(C)on4)=O)C)C3C2)=O)CC2OC(=O)OC2C1 14660,C12(C(N3C(CC(NOCC(N)=O)=O)CCC3)=O)CCCC1C2(F)F 14661,Cc1ccc2nc(C(N3CC(O)CC3CNC(C3(C)CC=CCC3)=O)=O)cn2c1 14662,C(=O)(CC(CC)C(C)(C)C)NCCCCNC(CC(C=C)CCC)=O 14663,N1(C(c2cn(C(C)C)nn2)=O)CC2=C(C1)CN(C(C1(c3cccs3)CC1C)=O)C2 14664,C(CNC(C1CC2(CSC2)C1)=O)(CC(F)(F)F)NC(C=NOC)=O 14665,CC(C)(C)C(CO)C(=O)N1CCCC1CCNC(=O)CC1C=CCC1 14666,n1(CC(=O)NC2C3CC(NC(C4CC4[N+](=O)[O-])=O)CC23)ncccc1=O 14667,C(C)(CO)(C(=O)N1CCCC(CN(C(=O)CCC2CCCC2)C)C1)OC 14668,C1(CCC(C)(C)NC(c2ncn(CC)c2)=O)CCCCN1C(=O)Cn1ccnn1 14669,N1(C(c2ccc(C#C)cn2)=O)C2CCC1CN(C(c1ncc(C)cc1OC)=O)C2 14670,C12(COC)CC(CNC(C3C=CCC3)=O)(CN1C(c1ccccc1CC#N)=O)C2 14671,C1(NC(c2scc(COC)c2)=O)CN(C(=O)CCC2(C)CC2)C2(CCCC2)C1 14672,C1(OC)CCCCC1NC(=O)C(C1CCN(C(C2CCNC2=O)=O)CC1)C 14673,O=S(CC(F)(F)F)N1CCCC(c2nc3ccccc3[nH]2)C1 14674,CN1C(=O)CCCC1C(=O)NCC(c1ccccc1F)NC(=O)C#CC1(C)CC1 14675,C1(NC(C(C(C)OC)O)=O)CCCN(C(=O)CN2CCN(C)CC2)CC1 14676,N1(CCC(=O)NCCC2(NC(C3OCC(C)C3)=O)CC2)CCC(O)CC1 14677,c1(C(=O)NC2CCN(C(C3C(CC)OCC3)=O)CC2)cc2c(s1)CCCCCC2 14678,C#CCC(O)C(=O)NCCC(=O)NOCCOCCOC 14679,C#Cc1cc(C(N2CCCCC2CNC(=O)C(O)Cc2cnc[nH]2)=O)ccc1Cl 14680,C1(CC(=O)NCCN(C)CC)CN(C(c2cn3c(n2)CCC3)=O)CCC1C 14681,C1(C(N2CCCC2C(F)(F)F)=O)CCCN(Cc2ncccc2Br)C1 14682,c1(C(=O)NC(CN(C(c2c(C(C)C)ccc(C)c2)=O)C)C)ccc([N+](=O)[O-])cn1 14683,c1(C(N(C(C)CNC(C2CCN(C3CC3)C2=O)=O)C)=O)c(F)cncc1Br 14684,c1(C(=O)NC(C)CCCNC(C2(F)CC=CC2)=O)cc(C(F)F)ccc1F 14685,C#Cc1cccc(NC(C2(NC(=O)COC(C)CC)CC2C)=O)c1 14686,c1(CC)ccc(C(N2CC(NC(c3cccc(O)n3)=O)C(SC)C2)=O)c(Cl)c1 14687,CCC(C)(CC)C(=O)NCC(C)(CO)NC(c1cnc(C(C)OC)s1)=O 14688,S(=O)(=O)(c1cccc(=NCC2CC(C)C2)[nH]1)NC1C(CCCC)CCC1 14689,c1(OC)ccncc1C(=O)NCC1(C(C)NC(c2cc(F)cs2)=O)CC1 14690,C1(OC)CC(C)CN(C(=O)CC(C)CNC(C2(F)CCOC2)=O)C1 14691,c1(OC)cc(C(=O)N=S(C)(=O)CCO)c2cnccc2c1 14692,CC1CN(C(c2ccnnc2O)=O)CC1NC(C1(Cl)CC1(F)F)=O 14693,C#Cc1cnn(C)c1C(=O)NCc1cc[nH]c1C(N1CC=CC(O)C1)=O 14694,C1(C(=O)NCCOCCN(C(CC(CCC)O)=O)C)CCc2nnn(C)c2C1 14695,N1(C(C(C)(C)CO)=O)CC2CC(NC(=O)CCc3cccc([N+](=O)[O-])c3)CC1C2 14696,c1(NC(C(C(C)C)NS(N(C)CC)(=O)=O)=O)cc(C(=O)OC)ccc1Cl 14697,c1(-c2cnc(NC(Cc3nc(COC)sc3)=O)s2)ccc(C(=O)O)nc1 14698,C1(C(=O)Nc2cc(-n3cc(C(C)(C)N(C)C)nn3)ncc2)C2C(=O)OCC12Br 14699,N1(C(c2c(CC)nco2)=O)CCC(NC(=O)CCOCC(F)(F)C(F)F)C(C)C1 14700,C1(C(N2C(CNC(COc3cn(C(C)C)nc3)=O)CC2)=O)CC1C1CC1C 14701,c1(C(=O)NCC(C2CC2)NC(=O)C=CBr)cc(Cl)ccc1F 14702,CC(C(=O)N1CCN(C(=O)CCC2CC2)CC1CCO)C(C)(C)C 14703,C1(C(N2CCC(NC(CC(c3cccc(F)c3)C)=O)C2)=O)CCCCC1N(C)C 14704,c1(C(C)C)cccc(C(=O)NC2CC(NC(c3ccc(C(C)C)o3)=O)C2)c1O 14705,c1(C(N2CCCC(C(C)=O)C2)=O)cc(F)ncc1NS(C)(=O)=O 14706,c1(C(=O)NCCC2(OC)CN(C(c3c(CC)csc3)=O)C2)cc(C)ncc1C 14707,C12(CNC(C(CC)N(C)C)=O)CCC(CC1)N2C(c1nncn1CC)=O 14708,Cc1sc2ncnc(NCC3CCCC(NC(=O)CCCOC(C)C)C3)c2c1C 14709,N1(C(CN(C(=O)OCC)C)=O)CCN(C(c2sc(C)cc2Cl)=O)CC1CCO 14710,c1(C(N(C(CC)CC(=O)NCCc2ncon2)C)=O)ccc([N+](=O)[O-])[nH]1 14711,S(=O)(=O)(c1cnc(NCc2ccsc2)c(Cl)c1)N1CCCC(C(F)(F)F)(OC)C1 14712,C(=O)(C(CC(C)(C)C)NC(c1cscc1C)=O)NCC(CC(=O)OC)O 14713,N1(C(c2ncc(C)nc2)=O)CCN(C(=O)C=CC2CCCC2)CC1CF 14714,CCC(C)CCC(O)CC(=O)NCC(C)NC(=O)C(C)(F)C(C)(C)F 14715,C(C1CCCN1C(=O)CC1CCC1)=CC(=O)NCCCc1cccs1 14716,N1(C(c2nn(C)c(F)c2)=O)CC=C(CC(=O)N2CCCC3(C=CCO3)C2)CC1 14717,N1(C(c2cnc(C)o2)=O)CCCN(C(=O)C=Cc2cn[nH]c2)CC1C 14718,c1(C(N(CCC(C)NC(C2CC(N(C)C)C2)=O)C)=O)cc(CO)[nH]n1 14719,CC1(CNC(=O)C(O)c2ccsc2)COCCN(C(c2cc(C#N)c[nH]2)=O)C1 14720,c1(C(N2CCOCC(NC(=O)CC3CCCC4CC34)C2)=O)cnc2occc2c1 14721,C#CCC(C)(C(=O)N1CC=CC(O)C1)NC(=O)CC1(C#N)CCCCC1 14722,c1(CC(=O)NCCCCCNC(C2CC2C(F)(F)F)=O)cc(O)cc(Br)c1 14723,Cc1nn(C)c(C)c1CC(N1CCC(O)(C(C)NC(c2c(Cl)nsc2Cl)=O)C1)=O 14724,C(C1CN(C(C2OCCC2C)=O)CC1C(=O)N(C)Cc1cscn1)=CC 14725,C(C(C(F)(F)F)OC)NC(c1scc(CNC(C(C)OCCCC)=O)c1)=O 14726,C1(C(N(CC)Cc2cncn2C)=O)C2C3CCC(C3)C12.C1(=O)C=CC(C)N1 14727,C(=O)(C1=CCC(C)(C)CC1)NC1CN(C(c2ccn(C)c2)=O)C(CO)C1 14728,C(=O)(C(C)C(O)C(C)C)NC(CNC(CN(C1CC1)CC)=O)Cc1ccccc1 14729,c1(OC)cc(C(=O)N(CCC(C(C)C)NC(C2CCO2)=O)C)c2c(c1)CCCC2 14730,c1(CCC(=O)N(CCN(C(=O)CNc2ncccn2)CC)CC)ccc(Cl)cc1 14731,C(C)(CO)(CC(C)C)NC(C1CCN(C(Cc2c(C)n(C)nc2)=O)CC1)=O 14732,Cc1c(C(N2CCC2CNC(=O)CCSc2ccccc2)=O)c(C(F)F)nn1C 14733,C1(C)(C(=O)NC(C)CC2CN(C(=O)Cn3cnc(=N)[nH]3)C2)CCC(C)(C)CC1 14734,N1(C(c2cccc(F)c2)=O)CCC2(CCN(C(=O)OCc3ccccc3)CC2)C1 14735,C#CC1(C(=O)N(C(CCO)C(F)F)C)CCN(C(c2c[nH]cc2C)=O)C1 14736,CC1=C(C(=O)NCC(C2CCCC2)NC(C2CCC(C)NC2=O)=O)CCO1 14737,C1(NC(C2(C)C(C(=O)OC)C2)=O)CC(NC(=O)CC2CCOC2(C)C)C(O)C1 14738,C(c1ccc(C2CC2)cc1)=CC(=O)NC1CCCCC1NC(C1(CCF)CC1)=O 14739,c1(C(=O)NC2C(OC)CN(C(C(F)OC)=O)C2)ccn2cnnc2c1 14740,CC1=C(CC(=O)N(C)C(c2ccccc2)C2CCOCC2)c2ccccc2C1 14741,C(=O)(CCCC(C)(C)C)N1CC(C)(CNC(C2C(C)C2C)=O)OCC1 14742,CC1(C)CC(NC(c2cccc(C(N)=O)n2)=O)CN1C(c1cnnc(O)c1)=O 14743,C(=O)(CC(C)(C)C(=O)NCC1C2CN(C(=O)C(CSC)OC)CC12)OC 14744,N1(C(COC(CC)(C)C)=O)CCOC(C)(CNC(c2ccc(C)cc2F)=O)C1 14745,C1(NC(c2c(C)noc2N)=O)CC2(C1)CN(C(=O)C(c1cccc(Cl)c1)(C)C)C2 14746,CC(C)(C)CC(O)C(=O)NCCCCCNC(C1CCCCC1C(C)(C)C)=O 14747,c1(OC)nccc(C(=O)NC2CC(N(C(=O)C(C)N(C)C)C)C2)c1Br 14748,C(=O)(CCCC#CC)NCC(CC=C)NC(=O)C(c1ccccc1)F 14749,N1(C(CNC(CC)=O)=O)CC(CNC(=O)Cc2ncccc2C)CC1(C)C 14750,Cc1cc(C(N2CCOC(C(C)NC(C3(C#N)CC3C(F)(F)F)=O)C2)=O)nn1C 14751,C(=O)(C(F)(F)C(C)(C)O)NCC(C1CCN(C(=O)C(C)(C)CO)CC1)C 14752,N1(C(CC(CC(C)(C)C)O)=O)CCc2sccc2C1CNC(C1CC(F)(F)C1)=O 14753,c1(C(=O)NC2(C)CCN(C(CCc3ccc(C)s3)=O)C2)ccc2c(c1)C(C)CO2 14754,C(CCN=c1[nH]ccc(=NC2CCc3c(Cl)cccc32)[nH]1)N1CCCN(C)CC1 14755,C(c1ccc(OC)cn1)=CC(=O)N(C1CCN(C(C2C(OCC)C2C)=O)C1)C 14756,N1(C(C(C(C)C)NC(C)=O)=O)CCC(C)C(NC(c2snc(Cl)c2Cl)=O)C1 14757,CC(O)(CC(=O)N1CCCCC1CCCNC(c1cc(Br)c[nH]1)=O)C(F)(F)F 14758,C1(CNC(c2n(C(C)C)ncc2)=O)CN(C(=O)CN2C(=O)CCC2=O)C2CC12 14759,c1(CN2C(CCC(=O)Nc3ncc(Br)cc3I)CCCC2)cc(F)ccc1Br 14760,S(=O)(=O)(c1ccc(C)c(C)c1)NCC(=O)NCCNC(c1c(SC)cnn1C)=O 14761,c1(NC(N2CCOC(C(F)F)C2)=O)ccc(-c2cnco2)cc1 14762,N1(C(C2C(=O)NCC2)=O)CC2CN(C(=O)C=CC(F)(F)F)CC(F)(F)C2C1 14763,c1(CC(=O)NC(C)C(C)(C)NC(c2ccc(F)cn2)=O)cn2c(n1)CCCC2 14764,Cc1cc(N2CCCC(CCF)C2)ncc1S(=O)(=O)N1CCOCCC1C(C)C 14765,c1(OC)cncc(CCC(=O)N2CC(N(C)C(c3ncoc3CSC)=O)C2)c1 14766,N1(C(c2c(N)nccn2)=O)CCC2(NC(=O)C3=CCCCC3)CC2C1 14767,C1(C(=O)NC2CCCC(CC(=O)N(CCCCCO)C)C2)(CC)CCNC1=O 14768,C#CC1CC2CCC1N(C(C(=O)NC)C(C)CC1CCOCC1)C2 14769,CC(C)C(F)C(=O)NC(Cc1ccoc1)C(=O)NC1CC2(CCC2)C1 14770,c1(C(=O)NCC(CO)NC(c2ccc(OC3CC3)nc2)=O)cnn2c1CCCC2 14771,C(CC(=O)NCCC1CC1C)(C(F)F)NC(C1(Cl)C(C(C)=O)C1)=O 14772,C1(CCC(=O)NC23C(CN(C(C(C=C)(F)F)=O)C2)C3)CCc2ccccc2C1 14773,C1(S(N)(=O)=O)(C(=O)NC(CCCC)CNC(=O)CNC(=O)C2CC2)CCCC1 14774,N1(C(C2(C)CCCOC2)=O)CCOC2(CCN(C(=O)C(F)F)C2)C1 14775,N1(C(c2c(C)nc(CNC(C3CC(C)CO3)=O)o2)=O)CCN(C)CC1C1CC1 14776,N1(C(C2C=CC(NC(C(CN(C)C)O)=O)C2)=O)CCC(O)CC1C1CC1 14777,C#CCC(C)(C(=O)Nc1cc(CO)ccc1C)NC(c1ccc(OC)nc1)=O 14778,c1(C(=O)NC(CC=C)CNC(=O)CNC(c2cccs2)=O)cc([N+](=O)[O-])oc1C 14779,c1(OC)ccc2c(C)c(C(N3CC(C(C)NC(=O)CCCC(N)=O)C3)=O)[nH]c2c1 14780,O=C(C1CCCn2cnnc21)N1CC2(CNC(=O)C(F)(F)C3CC3)CCC1CC2 14781,CC(C)(C)C(CNC(c1ccc2nccn2c1)=O)C(=O)NC1(CO)CC(F)(F)C1 14782,CC(CCCC(=O)NCC1(C#N)CCC1)NC(c1ccc(F)c(O)c1)=O 14783,Cc1nccc(C(=O)NC2(C(=O)NCc3ccc(Cl)o3)CCN(C)C2)n1 14784,C=CCCCC(=O)NC1(CNC(=O)CCN2CCCC(C(N)=O)C2)CCOC1 14785,Cc1ccc(C)c(C(=O)NC(C)C(C)NC(c2nccc(Cl)c2F)=O)c1 14786,N1(c2nnc(C(=O)OCC)s2)CCCC(C2CC2NC(=O)CC)C1 14787,Cc1ccc(CN2CCC(O)(C(=O)NCCC(C)CO)CC2)c(F)c1F 14788,Cc1ccc(NC(=O)NNC(=O)NC(O)(Cc2nn[nH]n2)C(F)(F)F)cc1C 14789,C=CCC(C)(CC)C(=O)NCCC1(O)CCCN(C(c2ccc(OC)nc2)=O)C1 14790,c1(NC(C=C)C)nc(N2CCc3nocc3C2)nc2c1ncn2C(C)C 14791,c1(OCC(=O)NC2CC(C)(NC(CC(C)CF)=O)C2)cccc([N+](=O)[O-])c1 14792,CC(C(=O)NCC1CC(NC(c2cc(CCCO)on2)=O)C1)C(C)(C)C 14793,C1(C(=O)NCC2(CC(=O)NC(C(C)C)C)CC2)COC(=O)N1C 14794,CSC1=C(C(=O)NCC2(NC(=O)C(C)(O)CCc3ccccc3)CC2)CCCC1 14795,c1(CC(=O)NC2CC(NC(=O)CCn3ccnn3)CC2O)c(O)ncnc1O 14796,c1(C(=O)NC2CCC(NC(c3cc(Br)c[nH]3)=O)C2)cccc2nscc12 14797,N1(C(C(CC2CCCC2)OC)=O)CCN(C(c2cnc(C)o2)=O)C(C(C)C)C1 14798,N1(C(COC)=O)CCOC2CCN(C(c3cccc(C4(F)CC4(F)F)c3)=O)CC12 14799,C(=O)(CCC(=O)NCC1(NC(C2SCC=C2C)=O)CCCCC1)OC 14800,c1(C(CC)=O)ccc(C(=O)NCC2CCCCN2C(C2CC(C)N(C)C2)=O)cc1 14801,CCCCN=c1[nH]c(CC(=O)Nc2cccc(OCF)c2)cs1 14802,c1(C(N(CCCNC(C(C)OC(C)(C)C)=O)C)=O)cc2n(c1)CCCC2 14803,c1(C2CCN(C(=O)NCC(c3ccc(C)s3)N3CCCC3)C2)ccc(F)cc1 14804,n1(CC(=O)NC2CCC2NC(=O)CC2(CO)CCCCC2)nc(O)ccc1=O 14805,c1(OC)cn(C)c(C(=O)NCCN(C(=O)CCCCC2CCCCC2)C)cc1=O 14806,N1(C(c2cc(C)nnc2)=O)CCN(C(=O)C(C)CC(F)F)CC1CC(F)(F)F 14807,C1(C(=O)NCC2CCN(C(=O)C(c3cccc(C)c3)C)C2)(CC)CCCCC1 14808,N1(C(c2ccc(C)cc2N)=O)CCCC(O)(CNC(c2cnncc2C)=O)CC1 14809,C1(C(=O)NCC2(OC)CN(C(C3(F)CCOC3C)=O)C2)C2CCC1(C)C2(C)C 14810,c1(C(=O)NCCC(C)N(C(CCCC(=O)OC)=O)C)cccc2c1CCO2 14811,CC1=C(C(=O)N(CCCNC(=O)C(F)n2ccnc2)C(C)C)C(=O)OC1(C)C 14812,C1(C(=O)NCCOCCOCCCNC(C2C(C)(C)C2)=O)CCCCN1N=O 14813,C1(C(=O)NCc2cc(C(=O)NCC(COCC)O)ncc2)C2C3CCC(C3)C12 14814,N1(C(C=CCOC)=O)CC(NC(=O)CC(C)C(C)(C)CC)C2(CCOCC2)C1 14815,C1(NC(CCCCC)=O)CC(F)(F)CC1C(=O)Nc1nn(C)cc1C(=O)OCC 14816,C(CC(C)(C)C(F)(F)F)N(C(C)C1CC1)CCN1CC(C)(O)C1 14817,c1(NC(=O)NC2(C(N(C(C)C)Cc3ccccc3)=O)CC2)cc(Br)ncc1C 14818,CCCCCC(=O)NC1CC1CNC(=O)CN(c1ccc(Br)cn1)C 14819,O=C1Cc2c(C(=O)NC3CCN(C(c4cnnc(Cl)c4)=O)CC3F)cccc2N1 14820,C1(NC(CC=C=C)=O)CCN(C(=O)Cc2ccc(C(N)=O)nc2)CC1C(=O)OC 14821,Cc1ccc(F)cc1C(N1CCC2CC12C(=O)NC1C2CC3C(C2)C13CO)=O 14822,C1(C(N(CC(CC)NC(=O)CN(c2ccncc2)C)C)=O)C(C)(C)C1(F)F 14823,N1(C(CC2CCCN(C(c3cccc(CC)c3)=O)C2)=O)CCC2CCC(C1)N2C 14824,N1(C(CCCC(=O)NCCC)=O)CCC2(CCN(c3cc(C)ncc3C#N)C2)C1 14825,C1(CC(=O)NC(CNC(CCOCCC)=O)C)C(=O)N(C)N=C1C 14826,C(CCN)(C(F)(F)F)NC(=O)NC(c1cc(C(C)(C)C)ccn1)C 14827,c1(C(=O)NC2CN(C(Cn3c(C)csc3=O)=O)CC2C)cnc2ccc(F)cn12 14828,N1(C(c2ccc(OCCO)cc2)C(=O)NC(CC)(C)C)CCOC2(CCCCC2)C1 14829,N1(C(c2c(CC)oc(C)c2)=O)CCC(NC(=O)C(F)C2CCC2)C12CCCC2 14830,C1(NC(CC(=O)OC)=O)CC(F)CN1C(=O)C(C)C1(O)CCC1 14831,C1(OC)CN(C(C2CC23CCCC3)=O)CC1NC(=O)C(C)(C)NC(=O)C(F)(F)F 14832,C1(C(=O)NC2(CC)CC(C)(C)C2)CN(C(=O)C=Cc2ccncc2)CC1C1CC1 14833,c1(-c2scc(C(=O)NC3CNCCC3(F)F)n2)cc(F)c(F)c(F)c1 14834,C1(S(C)(=O)=O)(CN=c2nc(-c3c(-n4c(SC)nnn4)cccc3)[nH]s2)CCCC1 14835,C12(C(N3CCC(N(C)C(C4CC=CCC4)=O)C3)=O)CC(C#N)(C1)C2 14836,c1(OC)nccc(C(=O)NC2COCC2C(=O)N(C(C)(C)C(=O)OC)C)n1 14837,C1(C(N2CC(C)(NC(Cc3c(C)non3)=O)C2)=O)CCCC(=O)N1C 14838,CC1CCN(S(=O)(=O)CC(=O)N(CCCN(C(=O)CC2(C(F)F)CC2)C)C)CC1 14839,C(C)(CNC(c1csc(C)n1)=O)(CNC(=O)C(C)=C(C)C)OC 14840,c1(NC(CC(C)SC)=O)cccc(C(=O)NC(=O)CNC2CC2)c1 14841,Cc1cccc(CS(=O)(=O)NCCN(C)CCNC(=O)C#CC(C)C)c1 14842,C(=O)(C(C)CN(C)C(C1CCC1C)=O)N1CC(CSC)C1 14843,c1(NC2CCN(C(C(C(C)(C)C)NC(C)=O)=O)CC2)nc(C)c([N+](=O)[O-])cc1Cl 14844,N1(C(C2CN(C)C(=O)N2)=O)CC2CCC(C(=O)NCC(C)(C)CO)(C2)C1 14845,C1(CNC(c2cc3cc(Br)sc3[nH]2)=O)CC2(CCOCC2)CN1C(=O)CO 14846,C(CC(=O)N(C1CN(C)C1)C)(C(F)(F)F)NC(C(CC(C)C)O)=O 14847,C1(CCOC)(NC(c2ccsc2Cl)=O)CCN(C(C2OCCC2C)=O)C1 14848,N1(C(C(C=C=C)C)=O)CCC2(CC1)CN(C(c1cnc3c(c1)COC3)=O)C2 14849,C1(CNC(CCOCCC)=O)CN(C(c2c(N)cc(C)cc2F)=O)CC(C)(C)O1 14850,N1(C(C(C)=CC=C)=O)CC(CC(=O)N(C)CCOCCO)CC1C 14851,C1(C(=O)NC2CC(c3ccccc3)(NC(C=CC=CCC)=O)C2)C2CCCOC12 14852,C(=O)(C1=NOC(CC2(O)COC2)C1)N(CC(C)O)CCNC(=O)CC(F)(F)F 14853,c1(C(N2CCC(NC(C(C)(C)CC(F)F)=O)C(O)C2)=O)cc(Cl)ccc1[N+](=O)[O-] 14854,C(=O)(C(CCC(N)=O)N(C)C)NCC1(CNC(C2C(C=C)OCCC2)=O)CCC1 14855,c1(CC)nn(C)c(CC)c1C(=O)NC1CN(C(=O)CC2CC3CC3C2)CC1C 14856,C1(NC(CC(C=C)C)=O)CN(C(=O)CC23CCCN2CCC3)CCC1F 14857,c1(OC)ccc(C(N2CC(CCNC(C3CCSC3)=O)C2)=O)c(OC(F)F)c1 14858,c1(C(N2CCC(CC#C)(C(=O)NC(C)CF)C2)=O)cccc2c1CCC2 14859,Cc1cc(C(=O)NC(CC2CCOCC2)C(N2C(C)CC2(C)C)=O)sc1C 14860,Cc1c(CC(N2CC(NC(c3cccnc3S)=O)CC2C)=O)sc2ccccc12 14861,c1(OC)ccc(Br)c(C(N2C3CCC2C(C(=O)NC24CC(F)(C2)C4)C3)=O)c1 14862,c1(NC)cnncc1C(=O)NCC(C)NC(c1cncn1-c1ccc(Cl)cc1)=O 14863,C1(CC(=O)NC23CC2CN(C(=O)C(C)(C2CC2)OC)C3)(OC)CCCCC1 14864,C(c1cccc(F)c1)=CC(=O)N(CCCNC(C1(C)CC2CC2C1)=O)C 14865,c1(C(=O)NC(C(C)C)CNC(=O)C=CCF)cc2cc(Cl)cnc2[nH]1 14866,CC1CCC(C)(C)N1C(=O)CNC(=O)C(C)(C)C.c12cnc(nc1)-n1cc-2nn1 14867,N1(C(CNC(CCCCC)=O)=O)CC(NC(=O)Cc2ccc(C)nc2)C2CC2C1 14868,Cc1ncn(C)c1C(=O)NOCc1cn(CC2CC(F)(F)CO2)nn1 14869,N1(C(C(CCC)C)=O)CC(NC(c2cnc(N(C)C)c(Cl)c2)=O)CC2(CCC2)C1 14870,CC1(C)CC=C(c2cc(C(N3CCNC(=O)C3)=O)cc3[nH]ncc23)CC1 14871,CCC(CC)C(C)C(=O)N(CC(=O)N(C1CC(O)C1(C)C)C)C 14872,c1(C(C)NC(C(N2CCC(C)C2C)c2c(CCCC)ccs2)=O)ccccc1C 14873,c1(C(=O)NC(C)CCN(C(=O)CCC2CCCCO2)C)ccnc2ccsc12 14874,C=C(C)C1OCCC1C(=O)NCCCN(C(=O)COCCCF)C(C)C 14875,c1(C(N(CC(C)NC(C2CSCCS2)=O)CC)=O)cnn(CCN(C)C)c1C 14876,CC(C)(CCC(=O)N1CC(NC(C2CCC(CN(C)C)O2)=O)C2(CC2)C1)[N+](=O)[O-] 14877,Cc1ccnc(O)c1C(=O)N(C)CC1CCN(C(=O)C(c2cnn(C)c2)C)C1 14878,c1(C(=O)NCC2CC(NC(CCC(C)(F)F)=O)C2)ccc2c(c1)CCCS2 14879,C(=O)(CC1OCCc2sccc21)N1CC(C)(NC(c2cc3sc(Cl)cc3[nH]2)=O)C1 14880,CC1OCCC1N=c1[nH]c(N2CCOCC2)nc(=NCC2CC(O)C2)[nH]1 14881,C1(OC)CCCC(CNC(C2C3CC3CN2C(=O)CC2(C)CCOC2)=O)C1 14882,c1(C2N(C(c3cc(C4CC4)no3)C(=O)NCCOC)CCC2)cccc(Cl)c1 14883,c1(CNC(=O)CC2CCN(C(C3(CC4CC4)CC(O)C3)=O)C2)ccncc1Cl 14884,Cc1cnc(NC2CCC(C3CC3)C2)c(S(=O)(=O)NCC2(C)OCCO2)c1 14885,c1(OC)ccncc1C(N1CC(O)(C(F)C(=O)NCc2nccnc2C)C1)=O 14886,c1(OC)ccc(C(=O)NC(C)(C)CCCNC(=O)C(C)C)nc1Cl 14887,C1(C(N(CCC(N2CCC(CC3CCC3)C2)=O)C)=O)CC2(CC2)CN1C 14888,c1(OC)cnc2ccccc2c1C(N1CC(c2nn[nH]n2)CC1C)=O 14889,CC1(C(=O)NCC2(F)CCN(C(C3CCC(=O)O3)=O)CC2)Cc2ccccc2C1 14890,c1(OCC(N2C(C(C)NC(C(C)C)=O)CCC2)=O)ccc([N+](=O)[O-])cc1C(N)=O 14891,O(C1CCCc2ccccc21)CCNC(CCC1(C#N)CCOCC1)=O 14892,C1(C(N2CC(O)(C(C(=O)NC3CC(N(C)C)C3)F)C2)=O)CCOC(=O)CC1 14893,CC#CCCC(=O)NCC1CC2CC2N1C(c1cnn(CC2CC2)c1)=O 14894,CCC(C)C(O)C(=O)NCCCCCN(C(=O)C(C)SC(C)C)C 14895,CCC(C)C(=O)C(=O)N(CCCNC(=O)C(N1CCCCC1)C)C 14896,C1(NC(C2OCCN(C)C2)=O)CC2CC1CN(C(=O)C(C)(C)C(C)(C)C)C2 14897,c1(C(N2CC(C)C(NC(=O)CC3(C)CC3)C2)=O)ncnc2c1c(Br)cn2C 14898,C1(NC(c2c(Cl)cc(C)s2)=O)CCOC12CCN(C(=O)C=Cc1ccsc1)CC2 14899,C1(CNC(C(C)=C2CCC2)=O)CCCCN(C(=O)CC(C)N(C)C)C1 14900,C(=O)(CCCCCC#N)N1CCC(NC(C(C)(O)c2ccccc2)=O)C(O)C1 14901,C1(C(=O)NC2C3CN(C(c4c(C)n(C)nn4)=O)C2C3)CC12CCS(=O)(=O)CC2 14902,Cc1cccc(CNC(c2c[nH]nc2CCNC(=O)Cn2cc(C)cn2)=O)n1 14903,c1(C(N2CCC(O)(CCNC(CCS(C)=O)=O)C2)=O)c[nH]nc1[N+](=O)[O-] 14904,Cc1ccc(C(N2CCC(C)C2C(N2CC3CC2(C(N)=O)C3)=O)=O)cc1C#N 14905,c1(C(N(C2CCN(Cc3cnc(-c4ccccc4)s3)C2)C)=O)cc(Br)ncc1Cl 14906,c1(CC)nc(N2CCCC(NC(c3cc(C)ccc3C)=O)C2)cc(C)n1 14907,C(N=c1[nH]c(N2CC3CCCC3C2)nc2c1SCC2)c1cnc(O)nc1 14908,C1(NC(CCC(C)O)=O)CC2CCCC(C1)N2C(=O)Cn1cnc(=N)[nH]1 14909,c1(C(=O)NCC2OCCN(C(CCCCSC)=O)C2)ccc2nncn2c1 14910,C1(CC(=O)NC2CN(c3cc(CC)ncn3)C(C)C2)CCC(C)(C)CC1 14911,c1(C2(C(N(C)CCNC(=O)CCC3CC3(C)C)=O)CC2)cccnc1Cl 14912,C(=O)(CCCC#Cc1ccccc1)NC1C(C)N(C(=O)C2=COCCO2)CCC1 14913,c1(C(N(CC(C)NC(c2c(CC)nn(C)c2)=O)C)=O)ccc(COC)c(F)c1 14914,CC(CC(N)=O)C(=O)NCC1=CCN(C(=O)C(C(C)(C)C)C2CCCCC2)CC1 14915,C#CC1(NC(=O)C(F)C(C)CNC(c2n[nH]c(=N)[nH]2)=O)CCC(C)CC1 14916,c1(C(C)=O)cc(C(N2CCOCC2CCNC(=O)C=C2CCC(C)C2)=O)oc1C 14917,C(=O)(C(C(C)C)NC(=O)OC(C)C)NCc1scc(C(=O)NCC(CC)OC)n1 14918,C1(CC)CCN(C(c2ccc(I)cc2)C(=O)NCC(F)F)C1C 14919,Cc1ccc(C(=O)NCCOCC(=O)NCCN2CCCC(C)C2)cn1 14920,C(=O)(C(COC)CC(C)C)N1CC2CN(C(CNC(CC)=O)=O)C2C1 14921,C1(NC(c2ncc(C)c(Cl)c2)=O)CN(C(c2cc[n+]([O-])cc2)=O)CC1N=[N+]=[N-] 14922,Cc1ccc(C(=O)NCC(C2CC2)NC(=O)CC(C)C2CC2)c(C2CC2)c1 14923,N1(C(C(CC)OCC)=O)CC=C(C(=O)N2CCCNC(=O)CC2)CC1 14924,C1(C(=O)NCC23C(CN(C(C4C(C)OCCO4)=O)C2)C3)CC2(C1)CC(O)C2 14925,N1(C(C2(OC)CCOC2)=O)CCC(C(N2CC(F)(CF)C2)=O)CC1(C)C 14926,O=C(C1CCCc2cncn21)NC1CCN(C(C2(F)CCC(=O)CC2)=O)C1 14927,S(=O)(=O)(CCC(=O)NCC1(CNC(c2cncn2C)=O)CCCCC1)N(C)C 14928,C(=O)(CC1OCc2ncccc21)NCC1C(C)(C)CCCN1C(=O)C1=CCCC1 14929,N1(C(c2c(C)nn(C)c2)=O)C(C(N2CCOC(C(C)C)C2)=O)CCC12CC2 14930,N1(C(C(C)NC(C)=O)=O)CC=C(CNC(C2(c3ccnc(Cl)c3)CCC2)=O)CC1 14931,C1(OC)CC(CO)(NC(=O)CCc2cn(C(C3CCCCC3)C)nn2)C1 14932,CC1CC(CNC(=O)CCc2cc[nH]n2)CN1C(=O)Cc1cccc(Br)c1 14933,N1(C(Cc2cc(C)[nH]n2)=O)C2CCC1C(C)C(NC(=O)Cc1cncnc1)C2 14934,c1(C(=O)NCC(n2cc(COc3ncccn3)nn2)C)cccc2nn(C)nc12 14935,c1(CC(=O)N(C)CC2OCCN(C(C(C=C)(C)O)=O)C2)cc(F)c(C)cc1F 14936,Cc1c(NC(c2cc(I)cs2)c2nnnn2C2(C)CC2)cccc1Cl 14937,C1(NC(=O)NCCc2ccc(F)c(Cl)c2)CCOC2(CCS(=O)(=O)C2)C1 14938,C1(NC(c2cccc(O)c2F)=O)CN(C(c2ccoc2)=O)CCC1C(F)(F)F 14939,C(=O)(C#CC1CCC1)NC1(C)CC(NC(=O)CCC2CC2(Cl)Cl)C1 14940,C(=O)(C1=C(Cl)CCCC1)NCCC(=C)CNC(c1cnn(-c2ccccc2)c1N)=O 14941,N1(C(C2(C#C)CC2)=O)CCOC2(CCN(C(c3cn(C)nn3)=O)C2)C1 14942,c1(C(=O)NC2CCCC(NC(C(CCC)(C)C)=O)C2)ccc2nccc(C)c2c1 14943,c1(C(=O)NCC(C)N(C(C23COCC2C3)=O)CC)cc(F)cnc1O 14944,C(C(F)CNC(C1CC(NC(=O)OC(C)(C)C)C1)=O)NC(COCC#C)=O 14945,C1(C2(O)CN(C(=O)COCCOCCO)C2)(CNC(C(CC)(C)F)=O)CC1 14946,CCC(C)CC(C(=O)OC)NC(c1ccnc(O)c1F)=O 14947,c1(C(N(C2CCN(C)CC2)C)=O)ccc2[nH]nc(-c3cccc4ccsc34)c2c1 14948,Cc1ccc(=N)[nH]c1C(N1CCCC(CCNC(c2nc(Br)c[nH]2)=O)C1)=O 14949,CC(CS(C)(=O)=O)C(=O)N1CC2(CC(NC(=O)Cn3cccn3)CO2)C1 14950,N1(C(C(C)(CO)NC(C2CCCSC2)=O)=O)CCC12CCCC2 14951,N1(C(C(C)Br)=O)CCCn2nc(C(N3CCC(O)C(F)C3)=O)cc2C1 14952,CC(CC(=O)NC1C=CCC(C(=O)NC(C)(CO)C2CCCC2)C1)CC(C)(C)C 14953,C1(NC(CN(C)C(=O)C2CC2)=O)CCC(NC(c2ccc(NC(N)=O)s2)=O)CC1 14954,C1(c2nnnn2C2CCCC2)(NCCC(C=C)(C)C)CCOC(CC(=O)OC)C1 14955,CC1CC(CCNC(=O)C=CC2CCC2)CCN1C(=O)C(=O)NCC1CC1 14956,c1(CCC)cc(C(=O)N(C2CCCN(C(C3(F)CCCC3)=O)C2)CC)c(C)o1 14957,N1(C(CC(C2CC2)NC(C(C)O)=O)=O)CC(CO)C(O)C1 14958,c1(C(N2CC=CC(C(=O)NC(CC)(C)C3CC3)C2)=O)cc(C#N)oc1C 14959,N1(C(c2c(C)cn(C)n2)=O)CCCC2C1CCN2C(C1CC1C(C)(C)O)=O 14960,CC(C)(F)CCC(=O)N1CCC(CCCCCNC(=O)Cc2csc(=N)[nH]2)CC1 14961,Cc1ccc(C(=O)NC2CC2CNC(=O)CCSc2csc(C)n2)nc1 14962,S(=O)(=O)(c1cccc(OC(C)C)c1)NC(c1cc(CC)oc1C)=O 14963,NC(=O)CS(=O)(=O)c1ccc(C(=O)NCC(O)CNC(=O)Cc2cscn2)cc1 14964,C(=O)(C#CC(C)C)NCCOCCN(C(C=COCC)=O)C 14965,C1(COC)CN(C(=O)CCOc2ccc(Cl)c(Cl)c2)CC12CCC2 14966,N1(C(C(CCNC(CNC(CC)=O)=O)O)=O)CCCC2C(O)CC12 14967,c1(CC(C)(C)C)ccc(C(=O)NCC2CN(C(c3ncccn3)=O)C3CC23)cc1 14968,N1(C(C=CC(C)(C)C)=O)CCCCC(C(=O)NCCNC(C2CC2C(F)F)=O)C1 14969,C(C(CNC(C1CCCOC1)=O)C(F)(F)F)NC(CCn1c(C)ncc1)=O 14970,N1(C(CCOCC#C)=O)CCCC1(C)CNC(c1ccc(Cl)cn1)=O 14971,C(=O)(C1=CC2CCCC12)N1CC(CNC(C(c2cncc(F)c2)C)=O)OCCC1 14972,C1(NC(CCc2cncc(OC)c2)=O)CN(C(c2sccc2F)=O)C(C)(C)C1 14973,Cc1ccc([N+](=O)[O-])c(C(N2CC3CC2CN3C(c2cnn(C(F)F)c2)=O)=O)c1 14974,c1(C(=O)NCC(CO)NC(CN2CCCC(CC)C2)=O)nc(Cl)c(=O)[nH]c1N 14975,C(=O)(C1=CC2CCCC12)N(CCCCNC(c1c(C)cccc1)=O)C 14976,C1(C(=O)NCCOCCN(C)C)CC2(CCC2)CN1C(c1cn(C)nn1)=O 14977,Cn1ncc(NC(=O)CCC(N)=O)c1-c1cn(CC2CCCO2)nn1 14978,CN1CC2CCN(Cc3cccc4c3COC4)C2C1 14979,c1(CCC(=O)NCCNC(CCc2c[nH]c(=N)[nH]2)=O)ccc(C2CC2)cc1 14980,c1(C(=O)NC)cccc(C(=O)NC2CC(CCNC(C3CCOC3C)=O)C2)c1 14981,C1(NC(c2ocnc2C(F)(F)F)=O)CCC(c2ccccc2)CC1 14982,c1(C(=O)NCC(CC)NC(C2CC(C3CCC3)C2)=O)c(F)ccc(OC)c1N 14983,c1(N2CCC(C(C)NC(CC(CC)CC)=O)C2)nc(C)nc2n[nH]cc12 14984,C1(C(=O)NCC(=O)NCCC)CC2(CCC2)CN1C(=O)CNC(C1CC1C)=O 14985,Cc1ccc2ncc(C(=O)NCC(C(C)C)NC(=O)CN3CC(C)C3)c(=O)n2c1 14986,c1(NCC2(CC)CCCCCC2)cc(=NCC2CC3(CC3)CCC2O)[nH]c(C)n1 14987,CCCCCC(O)C(=O)NCCC(C)(C)NC(=O)Cn1cncc1C(=O)OC 14988,C#Cc1ccc(C(=O)NC2CC3(C(N4CCCC(C)(CC)C4)=O)COC2C3)cc1 14989,C1(C)(OC)CCCN(C(=O)C(C)(C)CCCNC(C2CC(C)(C)CCO2)=O)CC1 14990,C(=O)(CCc1ccco1)N(C(C)C(=O)OC)C1CC(n2cccn2)C1 14991,c1(C(N2CC(C)CC(NC(CCCC(C)C)=O)C2)=O)nccc2c1NCCC2 14992,c1(C(=O)NCCC2CN(C(C3(C)CC(C)OCC3)=O)C2)cnc2c(ccn2C)c1 14993,C1(CNC(c2ccc(CC)c(CC)c2)=O)CC2(CCC2)CN1C(=O)CC(C)(F)F 14994,CCCC(CCC)C(=O)NCC1CCCN(C(C2CCC(OC(F)F)CC2)=O)C1 14995,c1(CC(CNC2(CCC)CNC2)C)ccccc1C(F)(F)F 14996,c1(C(=O)NCC(C)CNC(C2(C)CC(F)C2)=O)cccc2c1nc(O)n2C 14997,N1(Cc2ccc(OC)c(Br)c2)CC2CCC1CN2C(c1cocn1)=O 14998,O=C1C=COC2(CCN(C(c3cc(Br)c(Br)o3)=O)CC2)C1 14999,C1(N(C(c2c(CC)n(CC)nn2)=O)C)CCN(C(C2(F)CCCCC2)=O)CC1C 15000,C=CCCCC(=O)N1CC(O)(C2CCCN2C(=O)C=CCCC=C(C)C)C1 15001,c1(OC)ccc(Cl)c(CN2CCCCC2CNC(=O)CC2CCC2)c1 15002,Cc1nc(C)c(C(=O)NC2(CNC(=O)Cn3nnnc3-c3ccsc3)CCC2)s1 15003,N1(C(C(C(C)C)=O)=O)CCC2(CCCN2C(=O)CC2NC(=O)NC2=O)C1 15004,c1(CC(=O)NC(CCOC)CNC(=O)C(=O)N(C)C)cccc2nonc12 15005,N1(CC)CCOCC1CC(=O)NC1CC(N(C)C(c2cccc(C(C)C)n2)=O)C1 15006,CN1CCN(C)CC(C(N2CC(C3CN(C(c4cccc(O)n4)=O)C3)C2)=O)C1 15007,C1(CSCC)CCN(C(c2ccc(C(F)(F)F)n2C)=O)CC1 15008,CC1CCCN(C(c2ccc(F)c(F)c2)=O)C1CNC(C1CC(F)(CO)C1)=O 15009,N1(C(CC2C(CNC(C=C(C)C)=O)C2)=O)CC(C2=NOC(C)C2)C1 15010,N1(C(c2cccc(C(N3CCC(F)(CO)C3)=O)n2)=O)CCC2(CC1)N=N2 15011,C1(C(=O)NC(C)CCN(C)C)OCCC1CNC(=O)CC1CC1 15012,c1(N2C(CCCNC(c3cn(CC=C)nn3)=O)CCC2)cc(C)nc(COC)n1 15013,c1(C(N2C(C(=O)OC)CC2C)=O)cccc(CNC(=O)CC2CC(F)(F)C2)n1 15014,C1(C(N(CCCNC(=O)CCCN2CCCC2)C)=O)CCc2nncn2C1 15015,C(CCC(N)=O)(C(=O)NC1CC(F)(C(=O)OC(C)(C)C)C1)NC(c1cccs1)=O 15016,N1(C(c2c(CC)n(C)nn2)=O)CCOC(C)(CNC(=O)CC2CCOC2(C)C)C1 15017,C1(NC(C2C(OCC)C2)=O)CN(C(=O)CCn2cc(Br)cn2)CC2(CC2)C1 15018,N1(C(c2ccc(C#C)nc2)=O)CC(NC(=O)C(O)CN(C)C)CC2(CC2)C1 15019,C1(C)(C(N(CC(C)O)CCNC(=O)C(=O)NCC2CC2)=O)CCN(C)C1=O 15020,c1(-c2nc(C(Cl)(F)F)c3ncnc-3[nH]2)scc2c1OCCO2 15021,N1(C(C(C(CC)C)O)=O)CC2CCCC1C2CNC(=O)C1=CCOCC1 15022,C(CCNC(c1nnnn1C(C)C)CCc1ccccc1)(C(C)C)OCCOC 15023,N1(C(c2cccc(OC)n2)=O)CC(C(=O)NC(c2ccc(F)cc2)C)CC(F)C1 15024,C1(CN(C(=O)C=Cc2cc[nH]n2)C)CCCN(C(C2CCOC(=O)N2)=O)C1 15025,c1(C(=O)NC(CC)CNC(c2ccnnc2O)=O)cc(O)ccc1[N+](=O)[O-] 15026,C12(C(N(C)CC3C(C)C3)=O)CC(CN(C(C3(C#N)CC3)=O)C1)C2 15027,c1(OC)ccc(F)c(C(N2C3CN(Cc4cccc(C#N)c4Cl)CC23)=O)c1F 15028,C=CC1(C(=O)NC(C)CCN2CCCC2)CCN(C(C2CCOC2C(C)C)=O)C1 15029,c1(C(=O)NC2(C)CCCN(C(C3CCC(O)C3)=O)C2)cncc2c1CCC2 15030,C#CC(C)CN=C(NCc1ccccc1)N1CCC(c2ccc(F)cc2)C1 15031,Cc1cnc(-c2noc(C(C3(C)CC3)F)n2)nc1 15032,c1(OC)ccc(N(C)C(=O)Nc2cc(N3CCOC3=O)ccc2F)cc1F 15033,Cc1nn(C(C)(C)C)c(C)c1C(N1CC=CC(NC(C2(F)CC=CCC2)=O)C1)=O 15034,Cc1cc(F)ccc1NC(=O)C(=O)NCc1cccc(C(N)=O)c1 15035,C1(C(=O)NC2C(c3cn(CCCCCC)nn3)CCC2)CN(C)CC(C)O1 15036,C(=O)(N=c1ccc(SC)n[nH]1)c1cc(CC)ncc1 15037,Cc1cccc2cc(C(N3CC4(C3)CN(C(=O)C3CC3)CCO4)=O)nn12 15038,C1(NC(CC(=O)NCC#C)=O)CN(C(=O)C(C)(C)c2ccccc2)CC12CC2 15039,C1(C(C)C)(C(=O)N(C)CCc2cnc[nH]2)CCN(C(=O)COC(C)(C)C)C1 15040,C1(NC(C2(F)C(C)OCC2)=O)CC2(CCN(C(=O)C=Cc3ccccc3)C2)C1 15041,C1(NC(C=C(C)C(F)F)=O)CCC(N(C(=O)C(c2cnn(C)c2)C)C)CC1 15042,C(=O)(C1=NNC(C(F)(F)F)C1)N1CCC(CN(C(=O)CCC(C)(F)F)C)C1 15043,c1(OC)ccc(NC(=O)C(c2cc(C)ccn2)N2CCC(F)(COC)C2)cc1 15044,C1(C)(CNC(CC(OCC)OCC)=O)CCN(C(c2cc3occc3[nH]2)=O)CC1 15045,C=CC1CN(C(=O)C(C)NS(C)(=O)=O)CC1NC(c1nc(C)no1)=O 15046,c1(CCC)n[nH]cc1C(=O)NC1CC(O)C1CC(=O)NCCN1CC=CCC1 15047,N1(C(CCc2n(C)c(S)nn2)=O)CC(NC(C2C3(CC3)C23CC3)=O)C2(CCC2)C1 15048,c1(C(=O)NCCCN(C(=O)C(C)C2CC2)CC)cc(C)ccc1C1CC1 15049,C1(C(N2CCN(CC)C(=O)C2)=O)CC2(CCN(C(=O)Cc3cccn3C)C2)C1 15050,N1(C(C(CC(=C)C)C)=O)CCC(C2CC2NC(C2(O)CCC(C)(C)CC2)=O)CC1 15051,C1(C)(C(N2CCC3C(NC(C(F)=CC)=O)C32)=O)CC(c2ccccc2)=NO1 15052,N1(c2nc(N(C)Cc3ncc(CC)s3)nc(C)c2)CCCc2ccccc2CC1 15053,C1(CC)(NC(C2CCC(=O)C(C)C2)=O)CCN(C(C2CCC(=O)N2CC)=O)CC1 15054,c1(C(=O)NCCCNC(c2ccnnc2O)=O)ccccc1OCCF 15055,c1(C(=O)NC(CN(C(c2cc(=O)n(C)o2)=O)CC)C)csc2ccccc12 15056,c1(C(N2CC(CCC)N(C(=O)C=CC(=O)N(C)C)CC2)=O)c[nH]c2cccnc12 15057,N1(C(Cc2n(C(C)C)cnn2)=O)CC2(CC2)CC1CNC(c1nccn1C)=O 15058,c1(C(=O)NCCCCCNC(CCC(=C)Br)=O)cc2c[nH]nc2s1 15059,C1(CCNC(C(C)n2ccnn2)=O)CC(F)(F)CN1C(c1cc(Cl)cnn1)=O 15060,c1(CCC)nc(C(=O)NCC(O)C(=O)N(C)Cc2ccc(CC)o2)co1 15061,Cc1nn(CC(N2CCC(CO)C(NC(=O)CCOCC(F)F)C2)=O)c(C)c1Cl 15062,N1(C2CCN(C(C(CSC)OC)=O)C2)CCN(C(=O)CC2CCOCC2)CC1 15063,c1(C(N2C(C(C)(C)NC(C3CCC(C)C3)=O)CCC2)=O)cc2c(o1)CCCC2 15064,c1(C(N(C(CNC(C(C)NS(C)(=O)=O)=O)C2CC2)C)=O)sc(F)cc1Cl 15065,S(=O)(=O)(CCC(=O)NC(C1CCOC1)CNC(=O)C(F)(F)c1cscn1)NC 15066,CC1(C)CCCC2(CN(C(C3COCCO3)=O)C2)O1 15067,C(=O)(C(C)CC(F)(F)F)N(C)CC1N(C(C(COC)O)=O)CCC1 15068,C(C(C)CN=c1c(C#N)c[nH]c2ccc(Cl)cc12)NC(Cc1cc(C)nn1C)=O 15069,c1(C(=O)NC23CC(C(=O)NCC4CCC(C)CO4)(C2)C3)coc2ccccc12 15070,CN1CCCC(C(c2scc(CC(=O)NC(c3cccs3)=O)n2)=O)C1=O 15071,c1(OC)cc(N)c(C(=O)NC(C2CCCCC2)CNC(=O)COC(F)F)c(F)c1 15072,C(CO)(C(=O)NCC1C=CC(NC(C2CCC(C(N)=O)O2)=O)C1)NC(N)=O 15073,c1(CNC(=O)NC2(c3cccnc3)CCC2)ccc(CN2CCOCC2)cc1 15074,C1(C(=O)NC2(NC(=O)CC(=O)NC3CC3)C(C)C2)CCOC(C)(C)C1 15075,C(=O)(C1CCCn2cnnc21)N(CCNC(C1CN2CCC1C2)=O)CC1CC1 15076,c1(C(N2C(CC)C(C(=O)NCc3cc(=O)cc[nH]3)CC2)=O)cnc2cc[nH]c2c1 15077,C1(CNC(c2ccc3ncccn23)=O)CCCC(F)(F)CC1 15078,CC#CCCC(=O)NC1CN(C(c2cnc(C(=O)OC)s2)=O)CC1OC 15079,C1(CC)=NC(C)(C(=O)NCCCC(C)(C)NC(C2CC(O)C(F)C2)=O)C(C)=N1 15080,c1(C(=O)NCC(CC(C)C)NC(c2ccc(CO)c(F)c2)=O)ccc(N)c(Cl)n1 15081,C1(C(N2C(CCC#C)CCC2)=O)CN(C(=O)C(O)C(C)CC)CCN1C 15082,C1(C(N2CCN(C(CC(C)(C)O)=O)C(CCO)C2)=O)CC2CCC(C1)S2(=O)=O 15083,c1(C(N2CCC(OC)CC2)C(=O)NCCC)cnc2sc(Br)cn12 15084,c1(C(=O)NC23CCN(C(c4c(CC)noc4)=O)CC2C3)ccc2c(c1)SCCN2 15085,c1(C(CC#N)NC(=O)NCCCCN2CCOCC2)ccccc1 15086,C1(C(N(CCC)CCNC(=O)C(CC)(CC)CO)=O)Cc2cccc(C)c2O1 15087,C(N=c1[nH]c(=NCCc2nocc2C)[nH]c2c1SCC2)c1c(OC)cncc1 15088,CCCC(C)(C)C(=O)N1CC(CCNC(C2CCC2C(F)(F)F)=O)C(C)C1 15089,N1(C(c2nn(C)c(C(F)(F)F)c2Cl)=O)CCN(C(C2CCNC2=O)=O)CC12CC2 15090,C(C)(C)(C(C)(C)CO)NC(CCC1CCCN(C(CNC(=O)OC)=O)C1)=O 15091,c1(CC)nc2c(C)csc2c(=NCC2CCCN2C(=O)C(C)NS(=O)(=O)CC)[nH]1 15092,CCS(=O)(=O)CC(=O)NC1CC1CC1(OC)CCCN(Cc2ccccc2)C1 15093,N12CCCCCC1OC(CC1CC(C(=O)OC)C1)C2=O.C(C)(C)(C)OC(C)=O 15094,C1(N(C)C(c2cc[nH]n2)=O)CCCCN(C(C2CC(C)(C)O2)=O)C1 15095,C1(C(=O)NCC2(NC(CCCNC(C(C)(C)C)=O)=O)CCC2)C(Cl)(Cl)C12CC2 15096,N1(C(C2(C#C)CCC2)=O)CC(F)CC1CC(N1CC(C)(C(=O)OCC)C1)=O.CC 15097,c1(CNCCNC=O)cn(Cc2ccc(C(=O)NCc3cc(C)no3)o2)nn1 15098,CC(CS(C)(=O)=O)C(=O)NCC1(F)CCN(C(c2ccc3ncnn3n2)=O)CC1 15099,C1(NC(CSCC=C)=O)COC2(CCCN(C(c3ccc(N(C)C)cc3)=O)C2)C1 15100,C1(C(=O)NC2CCN(C(C)C)C2)CCN(C(=O)Cc2ccn(C)c2)C1(C)C 15101,S(=O)(=O)(c1c(Cl)cc(Br)cc1Cl)N1C2CN(C(c3c(F)cncc3F)=O)CC21 15102,N=c1[nH]nc(Cl)cc1C(=O)NCC1(CO)CCN(C(c2ccncc2F)=O)C1 15103,C1(CN(C(CCCOCC)=O)C)CN(C(=O)CC2(O)CCCOC2)CCO1 15104,N1(C(C(C)=C(C)C)=O)CCN(CCCNC(=O)C(C)C(C)O)CC1 15105,c1(C(=O)NCC(c2ccccc2)NC(C(CSC)OC)=O)ccc(N)c(Cl)c1 15106,N1(C(CNC(=O)OC)=O)CCC(C)(C)C(C(=O)NCc2nc(C3CC3)no2)C1 15107,C(=O)(C1=C(Cl)CCOC1)N1CCC2(C(C(N(C(C(C)C)C)C3CC3)=O)C2)C1 15108,C1(C(=O)NC(CC(=O)NC)C)(NC(C2C(C(=O)OC)C2(C)C)=O)CCCC1C 15109,CC1CCC(NC(=O)CCOCC(F)F)CN1C(=O)Cc1ccc(O)c(O)c1 15110,c1(C(=O)NC2CCCC2NC(C2CCCCC2O)=O)cnc2nccn2c1 15111,C12(OC)CCC(C(=O)NC3(C)CN(C(=O)C(F)(F)C(F)(F)F)C3)(CC1)CC2 15112,N1(C(C2C(C)OCCC2)=O)CC2(CC2)CC1CNC(=O)C1=NNC(C(F)(F)F)C1 15113,c1(C(C(=O)NCCCSC)N(C(CF)CF)C)cncc(Br)c1C 15114,N1(C(Cc2cccc(C#C)c2)=O)CC2CC(NC(=O)CCC3CC3CC)CC1C2 15115,N1(C(CCCC(=C)C)=O)CCOC2(C1)CN(C(C1CC(=O)N(CCOC)C1)=O)C2 15116,C1(N(C)C(c2ccc(F)o2)=O)CCCN(C(=O)CC(c2cccc(F)c2)O)C1 15117,N1(C(c2c(CC)noc2)=O)CC2(CNC(c3ccn(C)n3)=O)CC(F)(C1)C2 15118,C1(CCNC(C=C(CC)C)=O)(NC(=O)COC(F)F)CCC1 15119,C1(C(N(C(C)CO)Cc2ccccc2)=O)CN(C(C2CCC=CO2)=O)CCO1 15120,N1(C(C(CC)C)=O)C2CCC1CC(F)(CNC(=O)C=CC(F)(F)F)C2 15121,N1(C(C2COCCN(C(C3CN(C(C)C)C3)=O)C2)=O)CCC12CCCOCC2 15122,C(C1=CCN(C(C2(S(C)(=O)=O)CC2)=O)CC1)NC(C1(C)CC(C#N)C1)=O 15123,CCCCCC(F)C(=O)NCC1CCCC1NC(=O)C(C)COCC 15124,C1(CC=C)(C(=O)N(C)Cc2n[nH]c(C)n2)CCCN1C(=O)CCc1cn[nH]c1 15125,C1(N(C(c2c(C)ccc(C)c2)=O)C)CCCC2CN(C(=O)Cn3cnnc3)CC12 15126,c1(C(C(=O)NCCOCC)N(CC(C)(C)OC)C)cc(C(C)=O)cn1C 15127,N1(C(CC2C(C)C(=O)CC2)=O)C2CC1CN(C(c1ccc(CCF)cc1)=O)C2 15128,c1(C(=O)OCc2nn(C)c(Cl)c2)nc(Cl)c(=O)[nH]c1N 15129,C=Cc1ccc(C(=O)N(CCC(=O)NC2CCCCC2)CC)cc1 15130,CS(=O)(=O)c1ccccc1-c1ccc2c(C(=O)N=c3cco[nH]3)nsc2c1 15131,N1(C(C(C)OCC)=O)CC(F)(F)CC1CNC(=O)C(C)Sc1ccccc1 15132,C1(C)(C(=O)NCC(C2CC2)NC(C2(C(=O)OC)C=CCC2)=O)C(C)(C)C1(C)C 15133,N1(C(C2C(C(C)C)CCC2)=O)C2CCC1C(F)C(NC(c1cc(Cl)cs1)=O)C2 15134,c1(SC)ccccc1C(=O)NC1CC1NC(=O)C(C)(C)CO 15135,C1(NC(C2CC(n3ccnc3)C2)=O)CCN(C(c2ccncn2)=O)CC1CO 15136,c1(C(N2CCC(COC(C)=O)C2)=O)cc2ccc(-c3cnc(C)nc3)nc2[nH]1 15137,C(=O)(C(C)(C)CC(C)(C)C)NC1(COC)CN(C(c2ccnnc2C)=O)C1 15138,C1(CNC(C(C)NC(COC)=O)=O)CC2CC2N1C(c1ccc(C(C)=O)o1)=O 15139,c1(C(=O)NCCOCCCN(C)C(c2cnc(O)o2)=O)cc(Cl)ns1 15140,c1(Cn2cc(CS(CC)(=O)=O)nn2)ccccc1CNC(=O)CC12CCCC1C2 15141,Cc1cc(C(=O)NCC(C)NC(=O)Cc2sc(C)nc2C)c(O)cc1F 15142,C1(NC(c2ccc(OC(C)(C)C)nc2)=O)CCC2(CC1)CN(C(N)=O)CCO2 15143,c1(C(=O)NCC2(COC)CCCN2C(C2CC2(C)C)=O)cncc(N=[N+]=[N-])c1 15144,c1(N2CCC(C)C(F)(F)C2)nc2cc[nH]c2c(=NCC(C)(C)c2ccccc2)[nH]1 15145,C1(C(=O)OCC)CCC(c2nnnn2C)(NCC2(S(C)=O)CC2)CC1 15146,c1(N2CC3C(C)C3C2)nc2ccccc2nc1N(C)Cc1ccc(S(C)=O)cc1 15147,C1(NC(COC(C)=O)=O)CCN(CCNC(=O)CNC(=O)CC(C)(C)C)CC1 15148,C#CCC(C)C(=O)NCC1COCCN1C(c1ccc(N(CCCC)C)cc1)=O 15149,CCC(C(=O)NCCCCC1CN(C(=O)C(C)C2CCC2)C1)N1CCCC1=O 15150,CC(O)C(C(=O)NCCCCCCC1CC1)NC(c1ccc(O)cc1)=O 15151,c1(N2CC3CN(C(C(N4CCOCC4)C)=O)CC3C2)cc(Cl)c2cnn(C)c2n1 15152,c1(NCC(=O)N(CC(C)N(C)C(C2COCCO2)=O)C)cnn(C)c1 15153,C1(CC(=O)NCCC2(CNC(C(C)C)=O)CC2)CC(C(C)=O)C1(C)C 15154,N1(C(=O)C=CC2CCCC2)CCC(CCNC(C23CCC2CC3)=O)CC1 15155,C1(NC(C2(CC)CC2(F)F)=O)C2CN(C(C)=O)CC12 15156,C1(COC)(CNC(=O)C(CSC)OC)CN(C(=O)CC2(C(F)(F)F)CCC2)C1 15157,CC1(C)CN(C(c2csc(S(N)(=O)=O)c2)=O)C(CNC(=O)C(C)(C)C(F)F)CO1 15158,c1(C(=O)NC2CC(OCC(=O)NC3COCCC3(F)F)C2)ccc(F)c(F)c1 15159,S(=O)(=O)(c1cccnc1N(C)CC1CCCS(=O)(=O)C1)NCCN(C(C)C)C 15160,Cc1ccc(NC(=O)C(=O)NC2CCCC2C(C)C)c2ccccc12 15161,C(=O)(C(c1cccs1)=Cc1cccs1)NC(C(C)NC(C1(Cl)CC1)=O)C 15162,N1(CC)CCN(CCNC(N2CCCC(COc3cccc(SC)c3)C2)=O)CC1 15163,CC(CCNC(=O)CC1CCC1)CCNC(C1COCCO1)=O 15164,N1(C(C(CCC)O)=O)CC(C2CCCN(C(=O)Cc3cnc4cccnn34)C2)C1 15165,C1(NC(C(C2CC2)OCC)=O)CCC(F)(CNC(c2cc(C3CCC3)[nH]n2)=O)C1 15166,C1(F)(CNC(c2c(C)snc2)=O)CCCN(C(c2cnnn2C2CC2)=O)C1 15167,CCCCC(C(=O)NCc1ccc(C)cn1)NC(=O)C(C1CCCCC1)C 15168,CC1CN(C(C2CN(C(c3ccc(C#N)o3)=O)CC2(C)C)=O)CCS1=O 15169,N1(C(CS(CC)=O)=O)CCCN(C(c2cnc(C)nc2C)=O)CC1C(C)C 15170,c1(C(=O)NC(C)CC(C)NC(=O)C(C)CSC(F)(F)F)csc(=NC2CC2)[nH]1 15171,Cc1ccccc1Oc1ccc(C(N2CCC(N(C(=O)CC#N)C)CC2)=O)cc1 15172,c1(CC)onc(C)c1C(=O)NC1CCC(N(C(=O)CSc2n[nH]c(C)n2)C)C1 15173,CC1CN(C(=O)C=Cc2ccco2)CC(CCNC(=O)CCc2cncs2)O1 15174,C=CCCCC(=O)NCCC1(OC)CN(C(c2csnc2Cl)=O)C1 15175,c1(C(=O)NC(CC)CN(C(=O)CC2(CSC)CC2)CC)cncc(OCCO)c1 15176,c1(CC)cccc(C(N2CCCC(CNC(C3(Cl)CC3(F)F)=O)C2)=O)c1 15177,c1(NC(C2(F)CN(S(C3(CC=C)CC3)(=O)=O)C2)=O)cc(O)c2ccccc2n1 15178,C1(NC(C=CC(C)C)=O)CCN(C(=O)CCc2cc(Cl)no2)CC1C(C)C 15179,Cc1ncc(CNC(=O)C(CN(C)C)NC(=O)Cc2cnnn2C)s1 15180,C(C)(C)(C(=O)NC1CN(C(c2cn(Cc3ccccc3)nn2)=O)C1)SC 15181,C1(NC(C(CCCOC)C)=O)CCCCN(C(=O)Cc2cccc(C)c2)CC1 15182,Cc1cccc(C(N2CCCC(C)C2CNC(=O)CC2(CO)CCCC2)=O)c1O 15183,c1(C(N2CC(C)(CC(=O)Nc3ccc(I)c(Cl)n3)C2)=O)cccc2[nH]ncc12 15184,N1(C(c2cc(C)ncc2C)=O)CCCC(O)(CNC(=O)CCSCC(N)=O)CC1 15185,N1(C(Cn2c(=O)sc(C)c2C)=O)CC2ON=C(CNC(c3ccn(C)n3)=O)C2C1 15186,N1(C(c2c(C)nc(CC(C)C)o2)=O)CCC2(CC1)CC2NC(=O)CSCC(N)=O 15187,N1(C(CCOCc2nnc(C)s2)=O)CCCC(N(C)C(c2ccccn2)=O)C1 15188,N1(C(c2c(C)ccs2)=O)CCC(=CCNC(C2CC(F)C(=O)N2)=O)CC1 15189,C1(OC)CN(C(=O)C(C)=C2CC2)CC1NC(c1ccc(F)s1)=O 15190,Cc1cc(COCC(=O)NC2(C)CN(C(C3CCCN3C)=O)C2)on1 15191,N1(C(C2(C)N(C(c3c(C)cno3)=O)CC2)=O)CC2CC(C1)c1ccccc12 15192,Cc1cc(C(=O)NC2CCN(C(C3(C)CC3)=O)CC2C)c(C)n1-c1cnn(C)c1 15193,C1(C(N(C2CCN(C(C(C)OC3CCCCCC3)=O)C2)C)=O)CCCCS1(=O)=O 15194,C12(NC(=O)CCCc3cccnc3)CC(C1)N(C(c1cc[nH]c1)=O)C2 15195,C1(C(=O)NC(C(=O)NCC)CC)CCN(C(c2cc(C)n(C)n2)=O)C1CC 15196,C(C)(C(=O)NNS(=O)(=O)c1cc(C(F)(F)F)nn1C)Oc1cccc(C)c1C 15197,C(CCC(CO)NC(c1coc(C2CC2)n1)=O)NC(=O)CCCF 15198,c1(OC)cc(OC)[nH]c(=NCC2(C)CCN(C(=O)C=C3CCSCC3)C2)n1 15199,Cc1cccc(O)c1C(=O)NC1CC(CCC(=O)NCc2cn(C3CC3)cn2)C1 15200,N1(C(C(CC)OC2CCCC2)=O)CCCC(CC#N)C1 15201,c1(OC)cnc(Cl)[nH]c1=NC1CCCN(C(c2coc(CC3CC3)n2)=O)C1 15202,C1(C(=O)NC(CSC)(C)C(=O)N2CCOC(C(C)C)C2)CC2(CC(=O)C2)C1 15203,C(C(CC(C)C)C(=O)Nc1cnn(C)c1C(F)(F)F)OC 15204,C1(CNC(CC2(C)CC2(F)Cl)=O)CC2CCC1N(C(c1ccn(CC#N)n1)=O)C2 15205,CCCCCS(=O)(=O)NC(=O)CC(F)(F)c1cccnc1 15206,Cc1c(C(=O)NCC(C)N(C)C(C2CC(F)(F)C2)=O)cnn1C(C)(C)C 15207,N(C1C(=O)Nc2cccc(C)c21)C(c1ccc(-c2ccc(C)cn2)cc1)=O 15208,N1(C(c2ncn(C)n2)=O)CC2CC2C1CNC(c1cncc(O)c1)=O 15209,c1(NC(NOCCS(C)(=O)=O)=O)ccc(Cl)c(C(=O)NCc2ccco2)c1 15210,N1(C(c2cc(Cl)c(C)cc2Br)C(=O)NCCOC)C(C)C2CCCCC2C1C 15211,CC1(C(=O)NCC2(CNC(c3ccc(F)c(Cl)c3)=O)CCC2)CCCCNC1=O 15212,c1(CCC(=O)NC2(CO)CN(C(C(CC=C)C)=O)C2)ccc(Cl)c(C)c1 15213,CCCCCCCCCNC(C1CCN1C(c1c(F)cc(OC)cc1F)=O)=O 15214,c1(C(=O)NC2CC(NC(C(CC=C)C)=O)CC2O)ncc(F)c(OC)n1 15215,c1(C(CNC(C2CCCSS2)=O)NC(C(CC)OC)=O)ccc2ccccc2c1 15216,c1(C(N2C(CNC(CSCC)=O)COCC2)=O)c(Br)ccc2cccnc12 15217,Cc1ccc(-c2cc(CN3C(C)C(=O)NCC3)on2)cc1.C(N)(=O)NC 15218,c1(C(=O)NCCC2CCC(NC(C3(C=C)CCC3)=O)C2)ccc(C#N)cc1 15219,C(=O)(C=CS(C)=O)NC(C1(O)CN(C(=O)C(F)(F)c2cscn2)C1)C 15220,CC1(C)CCCc2c1n[nH]c2C(N1CC(NC(c2occc2F)=O)C1)=O 15221,c1(CC(=O)NC2(C)CC(C(N(CC(=O)OCC)CC)=O)C2)cccc(F)c1 15222,N1(C(C(C)CC2CCC2)=O)CCC(CO)(CNC(c2c[nH]cc2C2CC2)=O)CC1 15223,C1(C(N2CCSC2C(F)(F)F)=O)CC2CCC(C1)S2(=O)=O 15224,Nc1cc(C(N2CCCC3(NC(C4CC=CC4)=O)CC3C2)=O)cc(F)c1O 15225,C1(c2cccnc2)(C(N2CC(NC(C=CCC)=O)C2)=O)CCCC1 15226,C1(NC(C2(CC#C)CCCC2)=O)CCC(C)N(C(c2ccc(Cl)cc2N)=O)C1 15227,c1(CNC(C2CSCCN2C(c2cc(F)c[nH]2)=O)=O)ccccc1F 15228,c1(C(N2CC(COC)(CNC(=O)CC=CC(C)(C)C)C2)=O)ccc2cc[nH]c2c1 15229,C1(CNC(c2scc(C)c2)=O)CC2COCC2N1C(=O)C(C)CN(C)C 15230,C1(NC(C=CC(=O)NCCC(C)N(CC(F)F)C)=O)CCCCCO1 15231,CC(c1cnn(C)c1)=CC(=O)NC1CCC(NC(C2CCN(C)C2C)=O)C1 15232,C#CCCC(O)C(=O)N1CCN(C(=O)COCCCC)CC1C(F)F 15233,c1(C(=O)NC2CC(C)(NC(C(CC)NC(N)=O)=O)C2)cnn(C)c1Br 15234,C1(CCN(C(c2sccc2Cl)=O)CC2CCCCO2)CCCN(C(=O)CSC)C1 15235,C1(CNC(C=C(C)Cl)=O)CC2CCC1N2C(=O)Cc1cccc(F)c1 15236,N1(C(CN2CCC(OC)C2)=O)CC(NC(=O)C(O)CN2CCCC2)CC1(C)C 15237,N1(C(C2C(C(=O)OC)C=C2)=O)C(C(=O)NCC(O)CN(C)C)CC1C 15238,N1(C(CC(=C)C)=O)CCN(CCNC(=O)CC(F)(F)Cl)C(c2ccccc2)C1 15239,CC1(CCNC(c2csnn2)=O)CCN(C(C2OCCC2C(F)(F)F)=O)C1 15240,C(=O)(NNC(=O)CNC1CCC(CC)CC1)n1cc(C(=O)OCC)nn1 15241,C(CCN=c1ncc(F)c[nH]1)N(C(C1CC1CO)=O)Cc1ccccc1 15242,Cn1ccc(=NC(=O)C(CCC2CC2)NC(c2c[nH]c(=N)o2)=O)[nH]1 15243,C(C)(CC(C)NC(C1CC1(Cl)Cl)=O)NC(CSCCN(CC)CC)=O 15244,N1(C(C2CC(NC(C)=O)C2)=O)CCC(F)(C(N2CCNC(=O)C2)=O)CC1 15245,C1(C)(CNC(C(C(C)C)CO)=O)CC(F)(F)CN1C(c1cccn2cnnc12)=O 15246,N12CCC(CC1)C2=O.Cc1cc(N(C(=O)CCCF)CC(C)C)n[nH]1 15247,C=CC(C)(C)C(=O)NCC1CCN(C(=O)C(C(C)C)SCc2ccccc2)CC1 15248,N1(CCNCC)CCC(CC(CC2CCC3CC23)C(=O)OCC)C1 15249,C1(C(C)C)CCOC1C(=O)NCCOCCN(C)C(c1nnn(C)n1)=O 15250,C1(NC(C(CC)F)=O)CCC2CCN(C(=O)CCc3ccccc3[N+](=O)[O-])C12 15251,c1(N2CC=CC(NC(c3nn(CC)nc3C)=O)C2)ncc([N+](=O)[O-])cc1CO 15252,C1(CC(=O)NC(c2sccc2Cl)C)CCN(C(C2(c3ccncc3)CC2)=O)C1 15253,C(=O)(C(CCCC)C(C)C)NC(CCN(C(C(=O)NCC)=O)C)C(C)C 15254,C1(NC(CSCCCC)=O)(CC)CCN(C(=O)C(c2cccnc2)C)CC1 15255,c1(C(=O)NC2CC(CNC(C3N(CC)CC3)=O)C2)c(N)cc(F)cc1Cl 15256,C1(C(=O)NC2(CNC(C3CC(SC)C3)=O)CCOCC2)Cc2ccccc2N1 15257,C1(C(=O)NCC(CCCC)NC(C2(C)C=CCCC2)=O)CCC2(CC1)CC(=O)C2 15258,CC(O)(CC(=O)N1CC(O)CC1Cn1cc(CC2CCC2)nn1)c1ccccc1 15259,c1(SCC(N2CCN(C(c3cnccn3)=O)C3CC23)=O)nc2ccccc2[nH]1 15260,c1(C(N2C(CNC(CCCC#CC)=O)CCC2)=O)ccc(Br)c2cn[nH]c12 15261,c1(CNC2CCC(NC(CC3N(C(C)=O)CCCC3)=O)C2)ccc(F)nc1C 15262,N1(C(CC=C=C)=O)CCC2(CCCCN(C(c3cnn(C)c3F)=O)C2)C1 15263,c1(C(=O)NC2CCC(CNC(CC(=C)Br)=O)C2)nnc(O)cc1O 15264,c1(C(N2CCCC(N(C(c3ccns3)=O)CC)C2)=O)c(OC)cccc1O 15265,CC1CN(C(c2csc(=N)[nH]2)=O)CC1C(=O)NC(=O)COc1ccccc1 15266,c1(C(=O)NC2CCCC(NC(CC=CC)=O)CC2)cnn2c1CC(F)(F)C2 15267,c1(CSC)nc(-c2cn(C)nc2I)n(C2CCS(=O)(=O)C2)n1 15268,c1(C(N2CCn3nccc32)=O)cc2n(c1)CCC2 15269,C1(C(=O)NC(C(C)NC(C(C)CO)=O)(C)C)CCC2(CC1)NC(=O)NC2=O 15270,CCCC(C)(C)C(=O)NC1CC(NC(=O)C(C)SCC)C1 15271,Cc1cc(C(=O)NC(C)CCN(C)C(c2cc(C(C)C)no2)=O)n(C2CC2)n1 15272,C(=O)(C(O)CC(C)(C)C)NCC1ON=C(C(=O)NCC(C(C)C)(C)C)C1 15273,c1(-n2cc(CCCCNC(C(C)n3ccnc3)=O)nn2)cccnc1C(=O)O 15274,N1(C(C2OCC(C)C2)=O)CCC2(CCCN(CCc3ccccc3)C2)C1 15275,C1(O)(Cc2nc(O)n[nH]2)CN(CC(F)F)C1.C12CN(C1)NC2=O 15276,C(=O)(C1=NOC2(CCC2)C1)N(CC(CO)(CO)NC(Cc1c(C)con1)=O)C 15277,N1(C(C2(OCC)CCC2)=O)CC2(CCN(Cc3ccc(C)cc3)CC2)C1 15278,Cc1cnc(NC(C2CC(F)CN(C(c3nc(C)ncc3Br)=O)C2)=O)c(C)c1 15279,Cc1cc(C)c(C=CC(=O)NCC2CC(NC(C3CCOC3=O)=O)C2)cc1C 15280,Nc1nc(C(N2CCC(NC(=O)CC3(CO)CC3)C(O)C2)=O)ccc1[N+](=O)[O-] 15281,C(=O)(CC(C)CC(C)C)N1CCC(COC)(NC(C2(CF)CC2(F)F)=O)CC1 15282,C(=O)(C#CC1CCOC1)NCCC(CNC(c1c(C)n(C)nn1)=O)O 15283,c1(OC(C)C(=O)NCC2(O)CC(NC(C3OCCO3)=O)C2)ccc(F)nc1 15284,c1(C(=O)NCC2N(C(c3scc(COC)c3)=O)CC(F)C2)cccc2c1CCC2 15285,C(=O)(CCCCCN=[N+]=[N-])OCCC(C(=O)NCC(NN(C)C)=O)CCO 15286,C12(NC(=O)OC(C)(C)C)CCC(CC1NC(C13CCC(NCCl)(CC1)CC3)=O)C2 15287,c1(C(=O)NCC(C(C)(C)C)NC(C2CCC(=O)O2)=O)cnc2[nH]ccc2n1 15288,Cc1ccc2oc(C(=O)NC3CC4CCC(C3C)N4C(=O)CCC(F)F)cc2n1 15289,c1(OC)ccc(CN2CCC2C(=O)NCC2CCCN(C)C2)c(OC(C)C)c1 15290,C1(NC(c2ccc(C)cc2Cl)=O)CC2CCCC(C1)N2C(C1CCCN1N=O)=O 15291,CC1(C)CN(C(C2CC(F)(F)C23CC3)=O)CCS1=O 15292,C(=O)(C1=NOC(C(=O)NC2CCCN(C(=O)CC(C)(C)O)C2)C1)OC(C)(C)C 15293,C1(O)(C(=O)OC)CN(C(CC2C=CCC2)C(=O)Nc2ccco2)CC1O 15294,N1(CC(C)C)C(=O)NC(c2cccn2C2CC2)C2=C1C1(CCSC1)NC2=O 15295,C1(O)(C(C)CNC(C2CCCS2)=O)CCN(C(c2cnn(CC(F)F)c2)=O)C1 15296,CCC(CNC(C1CC(N(C(=O)Cc2cc(C)[nH]n2)C)C1)=O)CCO 15297,N1(C(C(C)(CO)NC(CC2(N(C)C)CCC2)=O)=O)CC23CCC2(COC3)C1 15298,C1(N(C(C(C)N(C)C)=O)C)CCCCC1NC(=O)C(O)COCc1ccccc1 15299,CC1(C)CC(NC(=O)C(C2CCCCC2)F)CN(C(=O)Cc2cc[nH]c2)C1 15300,c1(C(=O)NCC(CO)NC(c2csc(CO)n2)=O)cc(C(F)F)ccc1Cl 15301,CCCC(CNC(=O)CC1CCC(C)(C)O1)C(=O)NCC1OCCC1(C)C 15302,c1(C(N2CCC(C(CNC(C3C4CCCC34)=O)O)CC2)=O)cccc2cncn12 15303,C1(NC(=O)CSCCC(F)(F)F)(CO)CCCN(C(c2csc3nccn23)=O)C1 15304,C1(NC(CS(CC)=O)=O)CC2CC1CN(C(c1c(C)ccc(Cl)c1F)=O)C2 15305,CC1CC2CC(C(=O)NC(C3CCCC3)CNC(C3(C)CC3)=O)(C2)O1 15306,C1(C(CC(=O)OC)NC(=O)CSc2n[nH]c(C)n2)CCC(F)(F)CC1 15307,c1(C(N(CCCNC(C2(C)CC(C)C2)=O)C2CC2)=O)n[nH]c2cc(Cl)ccc12 15308,C(=O)(CC(C)(O)C(F)(F)F)NC(C1CCCN1C(=O)C=Cc1cccc(O)c1)C 15309,C(=O)(C(S(C)(=O)=O)C1CC1)N(CC(C)NC(C1CN(C(=O)C2CC2)CCO1)=O)C 15310,C1(C2CC2)(C(=O)NCC2CC(C(=O)NCCNS(CC)(=O)=O)C2)CCC1 15311,Cc1noc2nc(C(=O)NC(C)CCCCNC(c3cnc(Cl)s3)=O)ccc12 15312,C1(CC(=O)NCC(CC)(C)NC(=O)CC(C)COC)CCC=CCC1 15313,CC1CN(C(=O)CCC(=O)C2CC2)CCC1NC(=O)C(C1CCCCCC1)(C)C 15314,N(C(=NCCc1ccc(F)cc1)N1CCN2C(=O)OCCC2C1)CCC(=C)C 15315,C(CCOCCO)(C(=O)NCC1CC12CC2)NC(c1cnc(C)s1)=O 15316,C1(CC)C(NC(c2cn(CCC(C)C)nn2)=O)CCCN1C(C1CC(O)C1)=O 15317,O=C1CN(C(C2CN(C(=O)CC3CCCSC3)CC2F)=O)CCN1 15318,N1(C(C2N(C)C(=O)OC2)=O)CC2(CC(C(N3CC(F)CC3CO)=O)CO2)C1 15319,C12(NC(CCC3C(C#N)C3)=O)CC(CNC(C34CSCC3C4)=O)(C1)C2 15320,C1(C(N2CC(c3c(C)nn[nH]3)C2)=O)CN(C(c2cc(Cl)n[nH]2)=O)CCN1C 15321,c1(N(CC(c2cccc(I)c2)O)C)ccc(C#N)nn1 15322,c1(C(=O)NCC2(O)COC2)ccc2nc(-c3cccc4ccncc34)cn2c1 15323,c1(C(=O)NCCC(C(C)C)NC(c2c(CC)nn[nH]2)=O)cncc(Cl)c1C 15324,c1(C(N2CCCC(C)(C(N3CCC(CC)C3)=O)C2)=O)cnc2cc(Cl)ccn12 15325,CCC(C(=O)N1CC(O)CC1CNC(C1(c2ccccc2)CCC1)=O)C(C)C 15326,c1(OC)c(Br)ccc(CN2CC(C)CC2C(N2CC3C(CO)C3C2)=O)c1F 15327,C(=O)(C(C(C)CC(C)(C)C)N1CC2OCCOC2C1)NCC=C 15328,N1(C(C2=CCCC2C)=O)CC23CCCC2(C1)CN(C(C1(C(C)(C)O)CC1)=O)C3 15329,c1(CC)c(C(N2CCOC(CC(=O)NC3CCC(O)C3)C2)=O)cnn1C 15330,c1(CC(=O)N(C(C)CNC(=O)CC2OCCOC2(C)C)C)coc2ccccc12 15331,C1(NC(c2cc(C)[nH]c2C)=O)CC2CCC1C(NC(=O)CSc1ccccc1)C2 15332,CC(CNC(=O)COCc1cnoc1-c1ccoc1)(CO)NC(c1cccs1)=O 15333,c1(CCC(=O)NC2CCCC2CNC(=O)COC2CCC2)ccc(C(F)F)cc1 15334,C(C1=NOC2CN(C(c3csc(-c4cnc[nH]4)n3)=O)CC12)NC(c1cnsc1)=O 15335,c1(OC)ccc(Cl)cc1C(=O)NC1CN(C(C2CC(=O)N(C(C)C)C2)=O)CC1(C)C 15336,S(=O)(=O)(c1nc(C(=O)O)ccc1Br)N1CC2CN(C)CC2(C)C1 15337,C1(CNC(c2c(C)nn(C)n2)=O)CN(C(=O)Cc2ccc(O)nc2)C2CCN1C2 15338,c1(C(=O)NC(CCCCNC(c2ccc(CC)cc2)=O)C)n[nH]c2c1CC1CC21 15339,N1(C(c2ccc(CNC(C(C)C3CCCO3)=O)s2)=O)CCCC12CCOCC2 15340,CC1(NC(c2ccccc2CO)=O)CCCN(C(=O)CC2CCC3CC23)C1 15341,c1(C(N(CC(C)NC(=O)C(C)(C)N2CCCCC2)CC)=O)c[nH]cc(C)c1=O 15342,C(=O)(CS(=O)(=O)C1CC1)N1C(C2CCN(C(c3c(OC)cccc3)=O)C2)CCCC1 15343,c1(CC)cccc(CNC(C2CCCCN2C(C2(C)CC=CC2)=O)=O)c1 15344,C1(OC)C(OC)CN(C(c2ccon2)=O)C1CNC(C1(C)CC2CC2C1)=O 15345,c1(C(c2n(C)nnn2)NCC2CC3CC3C2)ccc(S(C)(=O)=O)s1 15346,c1(C(=O)NCC2C3N(C(c4ncn(C)n4)=O)C(CC3)C2)cn2cccc(Cl)c2n1 15347,c1(C(=O)NCCC(C)NCC2(C)CCC(=O)C2)ccnc2c1cnn2C 15348,C1(N(C(=O)C(COC)OC)CCC)CCN(C(c2cc(CC)ccn2)=O)CC1 15349,C(=O)(C1(Cl)CCCC1)NC1C(NC(c2ccc3c(c2)CC3)=O)CCC1 15350,C1(NC(C2CCCO2)=O)CN(C(C2CC(=C3CCC3)C2)=O)CC1CO 15351,c1(C(N2C(CNC(C3ON=C(CC)C3)=O)CC2)=O)cc[nH]c2nccc1-2 15352,CON(CC1CCCc2ccccc21)C(=O)CC(C)(C)C(=O)O 15353,C1(NC(C2C(C)CCO2)=O)CCSC12CN(C(C1CCCCC1N=[N+]=[N-])=O)C2 15354,C1(C(C)NC(C(C2CCCC2)NC(C)=O)=O)CCN(C(C2(O)CCOC2)=O)C1 15355,c1(OC)cc(O)ncc1C(=O)NCC1CCN(C(=O)CC2CC2(C)C)C(C)C1 15356,C1(C(N2CCC(C(CNC(C=CSC)=O)C)CC2)=O)CC2CCCCCC12 15357,C1(CCC)CN(C(c2cn(C)nc2C2CCC2)=O)CCN1C(=O)CCF 15358,c1(SC)ncc(C(=O)NCCC2CCN(C(c3cnn(C)c3N)=O)C2)c(O)n1 15359,Cc1cc(O)nc(C)c1C(N1CC2(CO)CC1(CNC(=O)C#CC(C)(C)C)C2)=O 15360,C1(NC(C(C2CCCC2)NC(C(CC(=C)C)OC)=O)=O)CCn2ncnc2C1 15361,c1(CC)cc(C)ccc1C(=O)NC(C1CCCCC1)CNC(=O)C(C)(O)C(C)C 15362,C1(C(=O)NCC(C)(CC(C)C)NC(c2c(CC)scc2)=O)Cc2ccccc2S1 15363,N1(C(CC(COC)(C)O)=O)CC2C3CCC(C2C1)N(C(=O)CCS(C)=O)C3 15364,N1(C(C=C(C)C(F)F)=O)CCCCC1c1n[nH]cc1C(=O)N(CC(N)=O)C 15365,C1(C(N2CCC(F)(CNC(=O)C(Cl)=CCl)C2)=O)Cc2ccccc2O1 15366,S(=O)(=O)(C1CCC2(CCCCC2)C1)NC(c1nn(C)cc1O)C 15367,c1(C(=O)NC2C(CO)CCN(C(c3c(C)cn(C)c3)=O)C2)ncn2c1CCCC2 15368,N(C(=NCCC(C)(C)O)NC1CC1C1CC1C)C(C)C1CC1 15369,Cc1ccc(C(=O)NCC23CCC(CC2)N3C(c2cc(F)cnc2O)=O)c(C)n1 15370,C(=O)(CS(=O)(=O)CC)N(C)OC(c1cnn(CCCC)c1CC)=O.n12cc(nn1)C2 15371,N1(C(CN(CCOC)C)=O)C(CNC(c2nc(Cl)ccc2F)=O)CC2COCC12 15372,c1(C(=O)NCC2C(NC(c3cn(CC=C)nn3)=O)C2)cc(OC)cc(Br)c1 15373,c1(N2CCC(=C)C2)nc(=Nc2cccnc2C)[nH]c2c1ncn2C 15374,C=C(C(=O)N1CCC(C(N)=O)C1)C1CCN(C(=O)OC(C)(C)C)CC1 15375,N1(C(CSc2nc(C)[nH]n2)=O)CCN(C(=O)CC(O)C2CCCC2)C2CCC12 15376,N1(C(c2n(CC#C)ccc2)=O)CCCCCC1CNC(=O)Cc1ccc(F)cn1 15377,c1(C(=O)NC(CNC(C(C(C)C)C)=O)CO)cc(N)cc2ccccc12 15378,c1(C(=O)NCCC(C)NC(C2CC23CC(O)C3)=O)cnc(C(F)F)nc1 15379,C#CCCN=C(NCCC(C)F)N1CCC(C2CC2)C1 15380,C#CCCCC(=O)N1CC(NC(C2(CC)CC2(F)F)=O)C(O)C1 15381,N1(C(C=C2CCC(C)C2)=O)CCCC(CCNC(=O)CCc2cncs2)CC1 15382,N1(C(c2ccc(CC)s2)=O)CCC(C(=O)N(C)CCN2CCCC2CC)CC1 15383,c1(C(N2CC(O)(CNC(CC3(C)CC3)=O)C2)=O)ccncc1Br 15384,C(C)(CNC(c1coc(C)c1)=O)(C(C)C)N(C(Cc1cn(NC(C)=O)nn1)=O)C 15385,c1(OC)ccc(NC(c2sccc2Cl)=O)c(OC(F)F)c1 15386,Cc1cccn2c(C(N3CCCC(NC(c4cccn4C)=O)CCC3)=O)cnc12 15387,C(=O)(CC(C)(C)CNC(C1CC=CCC1)=O)NCC1CCCC(C)O1 15388,N1(C(c2c(C)cn(C(C)C)c2)=O)CCN(C)C(CNC(c2n[nH]c(C)c2C)=O)C1 15389,C1(CNC(C(C(C)C)SC)=O)CN(C(=O)CC(C)(C)C)CC1(C)C 15390,c1(C(N2CCC(OCCNC(c3ncc(C)nc3)=O)C2)=O)cn2nc(C)sc2n1 15391,c1(OC)ccc(N2CCC(C(c3ccccc3Cl)OC)CC2)nn1 15392,C1(C(=O)NC2(CO)CN(C(c3c(CC)n(CC)nc3)=O)C2)CN(C)C(=O)CCO1 15393,C1(NC(C=CCN(C(=O)CC2CCSCC2)C)=O)C=CCCCC1 15394,C#CCC(C)(C(=O)N1CC(O)(CO)C1)NC(=O)CN(CC(C)(C)C)C 15395,C1(C)(C(=O)NCC(CNC(C(CC)C2CCC(=O)N2)=O)O)CC(C)(C)C1 15396,C(CCC(C)(C)C(=O)N1CCCC1CC(NCP(C)(C)=O)=O)OC 15397,N1(C(c2n(C(C)C)ccn2)=O)CC2C(CNC(=O)Cc3cn[nH]c3)C2C1 15398,c1(CC(=O)OC)cccc(CC(=O)NC2CCN(C(c3sccc3C)=O)C2)c1 15399,c1(CC(=O)NCCCCCNC(C2C(OCC)C2)=O)ccc(Cl)c(Cl)c1 15400,C1(CNC(CCCOCCC)=O)CN(C(=O)CC(C)(O)CCC)CCC1(F)F 15401,c1(C(N2CC(C)C(NC(=O)C(C)(C)CN(C)C)C2)=O)nc(Cl)ccc1F 15402,c1(C(=O)NC2(C)CN(C(c3c(C)ccc(OC)c3)=O)C2)cccc2nc(O)oc12 15403,c1(C(N2CCN(C(c3[nH]cc(CC)c3)=O)CC2)=O)c(Br)sc(C)c1C 15404,n1(CC)ccc(C(=O)NCC2(C(N3CC(CO)CC3C)=O)CC(C)(C)C2)c1C 15405,c1(N2CC(NC(C3CC4(CCC4)CO3)=O)CC(C)(C)C2)nc2cccc(F)c2s1 15406,C1(CNC(C(CNC(c2ccnc(O)c2)=O)OC)=O)CC2(CC2)C(=O)O1 15407,Cc1cc(C(C)(C)C(=O)NCC2(C)CCN(C(C3CCO3)=O)C2)ccc1F 15408,N1(C(C2CC=C(C)CC2)=O)CC2CC1CCC2NC(=O)CCc1cn(C)nn1 15409,Cc1nn(C)c2ncc(C(N3CC4CCN(C(=O)C(F)C(C)C)C4C3)=O)cc12 15410,n1(C(CC)C)nnnc1C(C(C)(C)OC(C)C)NCCCCCO 15411,C1(C(=O)NC2(c3cn(C)nc3)CC2)CCC2(CN(Cc3ccc(C#N)cc3Cl)C2)O1 15412,N1(C(C)=O)CCN(C(=O)NCC2COCOC2)C(C)C1 15413,N1(C(C=C(CCC)C)=O)CCCC2CN(C(=O)CCCOCCOCC)CCC12 15414,c1(CNC(C(=Cc2cn[nH]c2)C)=O)nnn(C)c1C(N1CCC(C)(CCO)C1)=O 15415,C=CCC(C)(CNC(C1CCCC1CNC(c1coc(COC)n1)=O)=O)CO 15416,N1(C(CCn2cc(C(C=C)(C)O)nn2)=O)CCN(C(C)=O)CC(C)C1 15417,C1(NC(C2CS(=O)(=O)C2)=O)C2CC3CN(C(=O)COc4ccc(O)cc4)C1C3C2 15418,CC1(CNC(c2cnc(Cl)s2)=O)CCCN(C(c2c[nH]ccc2=O)=O)C1 15419,C12(N(C)C(C3CCCC3O)=O)CCC(CN(C(=O)COc3cccnc3)C1)C2 15420,C12(C(=O)NCC(CNC(C(C)Cc3ccco3)=O)F)CC(C1)C(C(F)(F)F)O2 15421,c1(C(=O)Nc2ccnc(C(C)(C)C)n2)cn(CCO)c(=O)nc1O 15422,C1(C)(OC)CCN(C(C2CC3C=CC2CC3)=O)CC1 15423,C1(C#N)(C(=O)NC(CC(C)NC(C(C)OC)=O)C)CC1(C)C 15424,C#CCC(C)(CC)C(=O)NCc1csc(C(=O)N(CCCC(=O)NC)C)c1 15425,N1(C(c2cnc(C)s2)=O)CCC(C)C(NC(C2CC(n3cnnc3)C2)=O)C1 15426,N1(C(C(CC)=CC)=O)CCC(C)C1C(=O)NCC(F)Cl 15427,C(C(=O)NC1CC(C)(NC(c2ccon2)=O)C1)(C(C)C)n1ncc(C)c1 15428,C1(C(=O)NCCOCCOC)CCOC1C(N(CCC(=O)NC)CCO)=O 15429,O=C(CC(CNC(C1CCC2CC12)=O)C1CCC1)NCC1(Cl)CC1(F)F 15430,C1(CNC(=O)COCC2CCOC2)CC(F)(F)CN1C(=O)CC12COCC(C1)C2 15431,c1(CC(=O)NCCCN(CC)CC2CCC(=O)NC2=O)cn2cccc(C)c2n1 15432,C(=O)(C(C(C)C)NC(=O)C=CCl)NCCN(C(C(C)OCC=C)=O)CC 15433,c1(OC)ccnc(-c2cn(C(C)CNC(=O)CCc3cc(C)on3)nn2)n1 15434,Nc1c(C(=O)NCC(C2CC2)NC(C2(c3cccs3)CC2)=O)cccc1Cl 15435,Cc1cn2c(n1)C(C)CC(C(=O)NCC(C)(C)CN(C(=O)C1=CCCC1C)C)C2 15436,c1(CNC(CC2(N(C(C(C3CC3)SC)=O)C)CC2)=O)ccc(Cl)o1 15437,Cn1nc(C(=O)NC2CCOCC2C(=O)NCCc2cocn2)cc1F 15438,N1(C(CCC(=C)C)=O)CCOC2(CCN(C(c3cccc(Br)c3N)=O)C2)C1 15439,c1(CCC)nc(C(=O)NCC(C2CC2)NC(=O)CN(C)C)co1.C1(C)CC1 15440,N1(C(C(CCC)NC(=O)OC(C)(C)C)=O)CC(C(=O)O)CCC12CCC2 15441,C(CC(C)C)(C(=O)N1CCCC(N(C)C(c2[nH]ccc2C)=O)CC1)NC(=O)OC 15442,c1(CC(N2CC(CCn3cc(CC(C)(C)C)nn3)C2)=O)c[nH]ccc1=O 15443,c1(C2C(C(=O)NC3(CCNC(c4n[nH]cc4Br)=O)CC3)CC2)ccccc1 15444,c1(NC(c2c(-c3c(C)csc3)cncn2)c2ccccc2)ccc2cc[nH]c2n1 15445,CC(C)(C)C(CCO)NC(C1(CCNC(=O)C2=COCCC2)CC1)=O 15446,Cc1ccc(CCCCC(=O)NCCCC(C)NC(C2COCCN2C)=O)cc1 15447,C1(CNC(CCCOCC)=O)CC2CCC1N(C(C1(C)CCCS1(=O)=O)=O)C2 15448,C1(NC(c2c(C)ocn2)=O)CN(C(c2cc(Cl)cn2C)=O)CC1C 15449,c1(C(=O)NC2CN(C(C3N(C)CCOC3)=O)CC2F)cccc2nn[nH]c12 15450,C(=O)(CC(C)(C)N(C(=O)CC1CCC1)C)N(CC(C)C)C 15451,c1(OC)cccc(OC)c1S(=O)(=O)NC1CCCC1C(=O)NCc1cccnc1 15452,c1(C(N(C2CC(NC(CCCCCC)=O)C2)C)=O)cn(CC)c2ccccc12 15453,C1(NC(C(CC)SC)=O)CCCCN(C(=O)C(C)=C2CC2)C1 15454,CC(C)CC(CNC(c1cnn2ccccc12)=O)C(=O)NC1COCCC1(F)F 15455,c1(-c2c(OCC)cc(F)cc2)ccc2c(c1)CN(Cc1cc(Br)cc(Cl)c1O)C2 15456,C12(C(=O)NCC34CC(NC(c5c(OC)cncn5)=O)(C3)C4)CC=CCN1CCC2 15457,N1(C(c2nc(CC)oc2C)=O)CCC(C)(C)C(NC(c2cc(C)nc(O)n2)=O)C1 15458,C1(NC(c2occc2Br)=O)C2CN(C(=O)Cc3cccc(O)c3)CC12 15459,c1(C(=O)NC(CC)CNC(C2CCCC2(C)C)=O)cccc2c[nH]nc12 15460,c1(C(=O)NCC(=CC(=O)NC(CN(CCCC)C)C)C)cccc(C)c1N 15461,N1(C(C(C)C2CCOC2)=O)CC(NC(=O)C(C2(O)CCCC2)F)CC(C)(C)C1 15462,Cc1cccnc1C(CC(C)C)NC(=O)C(O)C(C)C 15463,N1(C(CSCC)=O)CCC(CNC(C2CCC23CCC3)=O)C12CCC2 15464,C1(CC)(CC)SCCNC1C(=O)NCc1ccc(N2CCCCC2C)cc1C 15465,Cc1nc(C(N2CCC(C3CCCCN3C(=O)Cc3cnc[nH]3)C2)=O)c(C)s1 15466,C12(CNC(CC3C(C)(C)CCCC3)=O)CCCC1N(C(C1CC1(F)F)=O)CCC2 15467,O=C1CC(CC(=O)NCC2(NC(C3CC3OCc3ccccc3)=O)CC2)CN1 15468,CCCCC(CN(C)C(c1cc(CNC(C2(C#N)CC2(C)C)=O)ccn1)=O)CC 15469,Cc1cc2c(cc1C)OC(C(=O)NC1CCCC1NC(=O)C(N)=O)C2 15470,n1(CC(=O)N(CCOCCNC(CC(CCC)C)=O)C)nc2ccccn2c1=O 15471,c1(CC(CC)C)nc(C2CCC2(F)F)n(-c2cccc(F)c2)n1 15472,Cc1cc(C(N2CCCC2Cn2cc(C(C)(C)C)nn2)=O)c(-n2cccc2)s1 15473,C1(NC(C(C)(O)C2CCC2)=O)CN(C(c2cnc(C(F)(F)F)nc2)=O)CCC1F 15474,c1(NC(c2cccc(CC)n2)=O)nc(C)ccc1OC 15475,CC1(C)CN(CC=O)C1.C1(C(=O)OC(C)(C)C)COCC1CNC(=O)C(F)CC1CC1 15476,CS(=O)c1ccccc1CC(N1CCC(N2CCNC(=O)C2)CC1)=O 15477,C(=O)(CCCC(=O)NC1CCC1C(N1CCOCC(C(C)C)C1)=O)OCC 15478,C1(C(=O)NC2C(NC(c3occ(C)c3)=O)COC2)CC2CCCC(C1)C2 15479,N1(C(=O)C(Cl)(Cl)Cl)CCC2(CC1)CN(S(=O)(=O)Cc1ccccc1Br)C2 15480,C1(F)(CNC(CC2N(CC)CCOC2)=O)CCN(C(=O)CN(C)S(N)(=O)=O)CC1 15481,c1(C(C(=O)NC(C(C)C)CNC(=O)Cc2ccc(Cl)s2)(C)C)ccnc(O)c1 15482,C(=O)(C(CC)C(=O)NC(CN=[N+]=[N-])C(=O)NC(c1ccc(C)cc1)C)OCC 15483,Cc1ccc(C(=O)NC2C=CC(CNC(c3csc(Cl)n3)=O)C2)c(N)c1F 15484,c1(C(=O)NC(COC)CC(=O)Nc2cccc(F)c2O)ccc2[nH]ccc2n1 15485,C(=O)(C1CCC(=O)c2cccn21)N1C2C(CNC(CC(C)P(C)(C)=O)=O)C(C2)C1 15486,c1(OC(C)C(=O)N2CC(NC(c3ccccc3SC(F)F)=O)C2)ccc(Cl)nc1 15487,c1(OC)ccc(C(=O)NC2CC(NC(=O)C(F)C(C)C)C(O)C2)cc1Cl 15488,N1(C(c2cn(CCC)nn2)=O)CC(NC(=O)C=Cc2cc[nH]n2)C(CO)C1 15489,c1(OCC(C)C)ccccc1C(=O)N(C)CC1(NC(C2CCOCC2)=O)CC1 15490,C1(CNC(C2C(C(N)=O)C2)=O)CCC2(CCC2)CN1C(C1(CC2CCC2)CC1)=O 15491,c1(C(=O)NC(C2CN(C(=O)C(C)(F)C(F)(F)F)CCO2)C)cc2n(c1)CCCC2 15492,C12(NC(c3c(COC)ncs3)=O)CC1CN(C(c1cc(Br)co1)=O)C2 15493,N1(C(C(C)Cn2cccn2)=O)CCN(C(=O)C(c2ccc(Cl)cc2)O)CC12CC2 15494,C1(O)(CC)CN(C(C2(CNC(=O)C(C)CC3CCCC3)CC2)=O)C1 15495,c1(NCC2(OCC)CCOC2)ccnc(O)c1 15496,C1(C(=O)NCC(CC)NC(=O)CCN(C)CC)CCc2nc(C)ncc2C1 15497,Cc1nnc(NC2CC(F)(CNC(=O)Cn3ccc(O)nc3=O)C2)nc1C 15498,c1(SC)ccc(O)c(C(=O)NCC2(O)CCCN(C(C3CC3C)=O)C2)c1 15499,C(CCN=C(NCC1CCSC1(C)C)N1CCN(CC2CCCO2)CC1)OC 15500,N1(C(c2ccc(CCC)cc2)C(=O)NCCCOC)CCC(F)(F)C(C)C1 15501,CN=c1[nH]cc(C(N2CC(OCC(=O)N(C3CCSC3)C)C2)=O)o1 15502,CCCCCCCCCC(C)CC(c1nnnn1C(C)C)NCCC1(C)COC1 15503,CN1CCC(C)(C(N2CC3(CNC(c4cscc4C(F)F)=O)CC2CO3)=O)CC1 15504,Cc1cc(C(N2CCN(C(=O)CSC(C)C)CC2C(C)C)=O)n2nccc2n1 15505,c1(OC)ccccc1C(O)C(=O)NCC(CNC(c1c[nH]nc1OC)=O)OC 15506,CCCC(C(=O)NCCCN(C(c1ccn2cccc2c1)=O)CC)C(C)C 15507,c1(C(=O)OCC)cc(CN(C2CCN(c3sccc3C#N)C2=O)C)oc1C 15508,CC1CN(CC(=O)N(C)CCC2CCCCC2)CCN1C(C1CCCCN1C)=O 15509,Cc1cnc(C)c(C(=O)NCC2CCCN2C(=O)C(C2CCCCCC2)C)c1 15510,c1(C(=O)NCCn2cc(C(N(CC(C)O)CC)=O)nn2)cc(C)n(C)c1 15511,C(=O)(C(CN=[N+]=[N-])NC(=O)CC1CC1)NC(c1ccccc1)C 15512,C(CCOCCO)(C(=O)NCC1(Cl)CC1(F)F)NC(C(N1CCNC1=O)C)=O 15513,N1(C(c2cc(OC)no2)=O)CC(C2CN(C(c3ccc(CC(C)C)cc3)=O)C2)C1 15514,N1(C(C=CCOC)=O)CCC(C(C)NC(c2cccc(-n3cnnn3)c2)=O)CC1 15515,Cc1c(F)ccc(NC(=O)C(=O)NC2CCN(C(=O)CN3CCCCC3)C2)c1F 15516,C(=O)(C(O)CC(F)(F)F)N(C)CC1CCCN1C(c1cc2n(n1)CCO2)=O 15517,c1(C(=O)NCC2(COC)CN(C(=O)C(O)C(F)(F)F)C2)ccc2oc(C)nc2c1 15518,N1(C(C2C(NC(c3cn(C(C)C)nc3)=O)COC2)=O)CCC(O)C(F)C1 15519,c1(C(=O)NC(C(=O)NC(CCC=C)C)COC)cc(O)nc(O)n1 15520,C#CC12CCC(C(N3C4CCCC3CN(C(=O)C(C)OCC)C4)=O)(CC1)CC2 15521,c1(OC)ccc(C)cc1C(=O)N(CCCNC(c1nnn2c1CCC2)=O)C 15522,C1(NC(CCOc2c(CC)cccc2)=O)CC(F)CN(C(=O)C(F)C2CCC2)C1 15523,S(=O)(=O)(c1ccncc1)NC1CCC(CC(=O)NC2CCC(F)(F)C2)CC1 15524,c1(CC)sc(C(=O)NCC#CCNC(=O)C(c2ccc(Cl)cc2)C)cc1C 15525,N1(C(CCCC(=O)NCCC)=O)CC2CC3CC2C1C3NC(c1coc(C)c1)=O 15526,c1(C(N(CCCCNC(C2(Cl)CC2(C)C)=O)C)=O)ccn2c1CCCC2 15527,C(CC(C)(C)NC(c1cc(C)cs1)c1nnnn1C1(C)CC1)OCC.C(C)(C)O 15528,c1(N2C3CN(C(C4CN(C)C(=O)C4)=O)C(C3)C2)ncnc2c1ncn2C1CC1 15529,Cn1nc(C(=O)NCC2COCC2NC(C2CCS2(=O)=O)=O)c2c1CCOC2 15530,c1(C(=O)NC(C2CCN(C(C3(CF)COC3)=O)CC2)C)ccccc1COC 15531,C1(CCNC(CCC2CCC(C)O2)=O)(Nc2nnnn2C)CCOCC1 15532,N1(C(CCC)=O)CCN(C(=O)C(c2cnn(C)c2)C)C(c2cccc(F)c2)C1 15533,C(N=c1[nH]c(=NCCC23CC(CO2)C3)[nH]c2c1CCC2)c1ncn(C)c1Br 15534,c1(C(N2C(C(=O)O)(CC)CC(OC)C2)=O)cc2scc(Cl)c2[nH]1 15535,N1(C(COCCOCCOC)=O)CC2(CC2)CC1CNC(=O)C(C)CC(N)=O 15536,CC(CNC(=O)CCn1cccn1)C(F)C(=O)NC1CCCC1 15537,C1(C(=O)NCC(CCNC(c2ccc(CO)s2)=O)O)CN2CCCN1CC2 15538,C1(C(N2CCC(CNC(C3CC(O)(c4cccnc4)C3)=O)C2)=O)CC2CC1C2 15539,c1(C(=O)NCC(CN(C(=O)Cn2ncn(C)c2=O)C)O)ccccc1C1(C)CC1 15540,N1(CCOC)CCOc2ccc(-c3cccc(-c4nn[nH]n4)c3)cc21 15541,c1(C(=O)NC(CC)CNC(=O)CC2(O)CCCC2)ccc(Cl)cc1O 15542,C12(CNC(C3CCN(C(C)=O)C3)=O)CCC1CN(C(c1cnccc1Cl)=O)C2 15543,Cc1oc(C)c(C(=O)NCCC2(c3cc[nH]n3)CC2)c1C.C1CCNC(=O)N1 15544,C(=O)(C1CCc2cccc(Cl)c21)N1CCC(NC(c2ccccc2F)=O)C(F)C1 15545,C1(CC)(CNC(=O)C(O)C2CN(C(C3(C)CC4CC4C3)=O)C2)CCCCO1 15546,N1(C(C2CN(c3ncc(OC)cn3)CC(F)C2)=O)CC2COCC(C1)C(=O)N2 15547,C1(C)(C(N2C(C(=O)NCC(C)S(N)(=O)=O)CC2)=O)CCC(=O)NC1 15548,N1(C(CN(C(C(C)C)=O)C)=O)CC=CC(NC(=O)CC2CCC(C)(C)O2)C1 15549,C1(NC(=O)CC2C=CCC2)CC(F)(CNC(c2cc(C(F)(F)F)cs2)=O)C1 15550,C(=O)(C1=CCC2(COC2)OC1)NC(CC)CN(C)C(c1nc(Cl)cs1)=O 15551,C(=O)(CCCC(=O)NC1CN(C(=O)C(O)Cc2cccc(Cl)c2)CC1O)NCC 15552,CC(c1ccco1)=CC(=O)NC1CCC(CNC(=O)CCN2CCCCC2=O)C1 15553,C(c1ccccc1Cl)=CC(=O)NCCC1CCCN(C(C(C)(C)OC(C)=O)=O)C1 15554,c1(C(=O)NCC2(O)CN(C(CC3CCCC(OC)C3)=O)C2)ccc2nsnc2c1 15555,CC1(C)CCC(C)(NC(=O)CC(CNC(c2cccnc2O)=O)C2CCC2)C1 15556,C1(NC(=O)NC(CC=CC)Cc2ccccc2)CC2CCC(C1)N2C 15557,CC1CCC=C1C(=O)NCC=CCC(=O)NOC1CCCC1 15558,C(=O)(CCC(=O)N(C(C)CNC(=O)CCCn1ccnn1)C)N(C)C(C)=O 15559,N1(Cc2ccc(C#C)s2)CCC2(CC(C(=O)NC3CCN(S(C)(=O)=O)C3)C2)C1 15560,C(c1ccncn1)=CC(=O)NCc1cc(C(=O)NC(C)CO)on1 15561,C(C(=O)NC1CCN(C(C2(F)CC=CC2)=O)C1)(C(C)C)OC 15562,c1(-c2ccc(CNC(C)(C)C(F)(F)F)s2)ccc2oc(O)nc2c1 15563,C(=O)(C(C)(O)C(C)(O)C(=O)OC)NC1(c2ccc(CC)cc2)CCC1 15564,c1(CC(=O)NCC#Cc2cn(C(C)C)nn2)nc2ccc(Br)cc2o1 15565,Cc1ccc(C(=O)N(C2CCN(C(c3cnc(O)o3)=O)C2)CCO)nc1O 15566,n1(C(C)C)cnc(C(=O)NC(C)CNC(=O)CCc2cc(Br)cs2)n1 15567,C#CCC(CC(=O)NC(C)C(C)(C)CO)NC(C1(CF)CC(=O)C1)=O 15568,C(CCN(C(=O)C(C)n1ccnc1)C)(C(C)(C)C)NC(CCOC(C)C)=O 15569,C(=O)(C(F)(F)CNC(C1CC(CNC(=O)CCN(C)CCO)C1)=O)OC 15570,N1(C(C2(C(C)NC(c3ccc(O)nn3)=O)CC2)=O)CCCN(C)CC1 15571,c1(COC)cc(CNC(c2ccoc2CNC(C2(C(C)C)CC2)=O)=O)no1 15572,c1(C(=O)NC2C(CNC(Cc3cc(C)sc3)=O)CCCC2)ccc2nccn2n1 15573,CC1(C(=O)NCCC2(O)CCCC2)CCCN(C(c2ccc(C#N)cc2)=O)C1 15574,C1(CC)C(NC(=O)C(C)CN(C)C)CCCN1C(C1CC12CC2)=O 15575,N1(CC(=O)NCC(c2cnccn2)C)CCCC(c2ccc(Cl)s2)C1 15576,CC1(O)CCCN(C(C2(NC(c3cc(Cl)c[nH]3)=O)CCOCC2)=O)C1 15577,C#Cc1ccc(C(=O)NCC(=O)NC(CO)(C(F)(F)F)c2ccc[nH]2)cc1Br 15578,c1(NC2CC(C(=O)OC)CN(C(=O)NCCO)C2)cc(Br)c(OC)cc1C 15579,c1(-c2scc(-c3c(C)cccc3)n2)ccncc1S(=O)(=O)N1CC2CC2C1 15580,N1(C(C(C=CCCC)O)=O)CCN(CCCNC(=O)C(C#N)CC)CC1 15581,c1(C(N2CC(O)(CNC(=O)CCCNC(=O)C3CC3)C2)=O)ccc(C(F)F)cn1 15582,C1(C(=O)O)CCC2(CCC2)N1C(C1CC(c2cccc(Br)c2)C1)=O 15583,CC1(C)CCN(C(=O)C2=CCCSC2)C1CC(N1CCOCC1)=O 15584,C12(C(C)C)COC(C(=O)NC(CNC(=O)CCc3cccc(Cl)c3)C(C)C)(C1)C2 15585,C1(C(=O)NC2C=C(C)CCC2)CN(C(=O)CN2CCNC(=O)C2)C2(CCC2)C1 15586,CCCC(C(O)C(=O)N1CCCC(C(C)(C)C)C1)NC(C1CCOC1C1CC1)=O 15587,N1(C(C2CC(NC(=O)Cn3cc(Cl)cn3)C23CCC3)=O)CCC(F)(F)C(F)C1 15588,c1(NCCN(CCCC)C)ccc(S(=O)(=O)NC(C)C(CO)SC)cc1Br 15589,O=C(C1=CCCOC1)NCC1CCN(C2CC2)C1.n12ccc(c1)C(=O)NCC2 15590,CCC(C)CC(CO)NC(=O)C(N1CCN(C)CC1)=O 15591,C(=O)(C(CC1COCCO1)C(F)(F)F)N(C)Cc1c(C)nn(C)c1C 15592,CC(N)CCCC(=O)N1CCC(C(N2CCC(c3ccc(F)cc3F)C2)=O)CC1 15593,Cc1cc(-c2cn(C(C)C(=O)NCC3CC4(CNC(=O)N4)C3)nn2)c(C)cc1Cl 15594,c1(C(=O)NC2C(CNC(C(CCC)F)=O)CCCC2)c(C)cccc1C 15595,N1(C(c2cc(OC)n(C)n2)=O)CC2CN(C(C3CC3F)=O)CC12 15596,CC(C)C(C#N)C(=O)NC1(C(=O)NCCC2CC=CC2)CSC1 15597,C1(O)(C(N2CCN(C(=O)CSc3ccc(Cl)c(F)c3)CC2)=O)CN2CCC1CC2 15598,c1(C(=O)NC(CNC(CSCCOC)=O)CC(C)C)ccc(F)c(Cl)c1 15599,N1(C(CCCCC=C)=O)CCC2C(C1)CN2C(C1CCN(CC(F)(F)F)C1)=O 15600,CCC(O)C(C)(C)C(=O)NC1C2CC1N(C(C1(NC(=O)CCC(F)(F)F)CC1)=O)C2 15601,Cc1cnc(C(=O)NCCC(=O)NCC2COCC(C)O2)cc1C 15602,C1(C(=O)NCc2cccc(C)n2)(COC)C=CCN1C(c1sccc1CO)=O 15603,c1(N2CCC(CCNC(=O)C(c3ccc(F)cc3)F)C2)ncnc(O)c1Br 15604,C12(c3n(-c4c(C)noc4C)nc(-c4cncc(F)c4)n3)CCCC(F)(C1)C2 15605,CC1OC(=O)NC1C(=O)NCC(C)(C)CCNC(=O)Cn1ccnn1 15606,C=CC(C)C(C)C(=O)NCC(C)(C)CNC(=O)CC1(CC(=O)OC)CCCC1 15607,C=C(F)C1(CC(=O)NC2CCCC(NC(C3(CO)CCCO3)=O)C2)CCC1 15608,N1(C(C2CCCC(C)C2)=O)CC2(CNC(c3coc(N(C)C)n3)=O)CCC1CC2 15609,c1(CC(=O)NCC2(F)CCC(NC(=O)CC3CC3)C2)ccc(O)c(Cl)c1 15610,c1(C(N(C2(C3CC3)CC2)C)=O)ccc(CCC(N)=O)cc1.C12(CCC1)C(=O)NC2 15611,O(N1C(=O)c2ccccc2C1=O)C(COC(C1CC2CCC(C1)S2)=O)=O 15612,N1(C(C(C2CC2)OC)=O)CC(F)(F)CC1C(=O)NC(C)CN1CCCCC1 15613,c1(C(=O)NC(CC(C)NC(CCOC)=O)C)ccc(C(C)=O)c(F)c1 15614,C#Cc1cncc(NC(C2C(CC)CCN2C(=O)C(C)CC2CCC2)=O)c1 15615,C1(CNC(CCSCC)=O)CCC2(CN(C(c3cc(N)c(N)cc3F)=O)C2)O1 15616,S(=O)(=O)(c1ccc(N2CCSCC(C)C2)c(C#N)c1)NC1C(CCC)C1 15617,c1(NC(C2CCCC(NCc3cccc(OC)c3O)C2)=O)c(O)cccc1C#N 15618,C1(C)(C(=O)NCCCN(C(=O)Cc2n[nH]cc2Br)CC)CCC(C)C1 15619,C1(CC(=O)NCC23CC(NC(C(c4cscn4)N(C)C)=O)(C2)C3)CC(O)C12CCC2 15620,c1(C(=O)NC2CC(CNC(C(C3CCOC3)OCC)=O)C2)scc2c1OCCO2 15621,C1(NC(C2C(OC)CCC2)=O)CN(C(=O)CN2CCC(F)CC2)CC(C)(C)C1 15622,c1(C(=O)NCC(CC)(C)NC(=O)C=Cc2cocn2)noc2c1CCCC2 15623,N1(C(c2cc(C3CC3)cs2)=O)CCCC(C2CC2NC(C2(n3cccn3)CC2)=O)C1 15624,CCC(C)(C)C(O)C(=O)NC1CC(C)CN(C(=O)C(F)(F)CN(C)C)C1 15625,c1(CC(=O)NC2C3CC(NC(C4C(CC)C4)=O)CC32)ccc2nc(C)[nH]c2c1 15626,c1(CC(=O)N(C2(C(=O)OC)CC2)C)ccc(CNC(C2CNC(=O)N2)=O)cc1 15627,N1(C(c2c(C)ocn2)=O)CCCC(NC(c2cc(=O)c(Br)c[nH]2)=O)CC1 15628,C1(C(=O)NCc2cc(C(=O)NCC3(Cl)CCC3)on2)(CC)CCCO1 15629,CCCC(C)(C)NC(=O)NC(Cc1ccccc1)C(=O)Nc1cccs1 15630,C#CCCCC(=O)NCC1C=CC(NC(c2ncsc2-c2ccccn2)=O)C1 15631,CCCC(F)C(=O)NCc1cccc(CNC(=O)C(F)CC)c1 15632,c1(CC(N2CC(Nc3ncnc(CC)c3F)C(C)C2)=O)noc2ccccc12 15633,CC1CCCC(O)(C(=O)NCCCCN(C(=O)COc2cnc(Cl)cn2)C)CC1 15634,Cc1nccnc1C(N1C(C(=O)NCC2(Cl)CC2(F)F)CCC1C1CC1)=O 15635,C(=O)(CCCCC(C)(C)OC)N1CCC(NC(CCCCC=CC)=O)(CC)CC1 15636,Cc1cc(C(=O)NCCC(C)(C)NC(=O)C(=O)N(C)C)nn1CC(F)(F)F 15637,CC1CC(CNC(=O)CN2CCCC2)CN(C(C2CCSC2)=O)C1 15638,c1(N2CCN(CC(=O)NC(COC)C)C(=O)C2)ccnc2cc(Br)nn12 15639,CCCC(CCCNC(=O)CCC(C)OC)NC(c1cc(F)ccc1N)=O 15640,c1(C(N2CC(C(C)NC(C(COC)(C)C)=O)OCC2)=O)n[nH]c2c1CCCCC2 15641,C1(CC(=O)NCCCC(C)NC(c2c(C)nsc2C)=O)CCCNC(=O)C1 15642,C1(C(=O)NCC2CCCCN2C(c2ccc(F)c(Cl)c2)=O)CC2(CCC2)CCO1 15643,O=S(=O)(c1c[nH]c2cc(Cl)ccc12)N1CC(O)(c2cscc2Br)C1 15644,C=C(C)CCC(C)(c1nnnn1Cc1ccco1)NC(CCC)CCCC 15645,N1(C(C2CC(=O)NC2)=O)CC2CCC1C(C(N1CCCCC1CCO)=O)C2 15646,Cn1cc(C#N)cc1C(N1CC(NC(=O)CCNC(=O)C=CCl)C(F)C1)=O 15647,C1(NC(C(CO)NC(C(CC#C)O)=O)=O)CCC(N=[N+]=[N-])CC1 15648,N1(C(c2nccc(C)c2)=O)CC(CNC(=O)CCc2cnc(C)o2)CC1(C)C 15649,CC1CCCCCC1Nc1cc(N2CCN(C(=O)N(C)C)CC2)ncn1 15650,c1(OC)cc(NC(C2CC(=O)N(C3CN(Cc4ccccc4)C3)C2)=O)cc(Br)c1 15651,CC1CN(C(=O)CC2CCCSC2)CC(C)N(C(c2cc(O)nc(O)n2)=O)C1 15652,C1(CC=C)(NC(=O)CN2CCCCC2C)CCN(C(c2cnn(CCF)c2)=O)C1 15653,C=C1CCN(C(=O)C(C)NC=O)C(C(=O)NC(c2ccc(C)cn2)C)C1 15654,N1(C(COCCOC)=O)CCC2(C)CN(C(=O)CNC(=O)C(F)(F)F)CC12 15655,CCCCC(C(=O)NCC(C)(C)C#CC(=O)NC1CC(CCF)C1)C(C)C 15656,C1(CC(N2CCCC2C2(C(=O)NOCCCCC3CC3)CC2)=O)COCCO1 15657,C1(NC(COC(C)=O)=O)CCCC2CN(C(c3ccc4cccnc4n3)=O)CC12 15658,C(=O)(C(O)CCC(F)(F)F)N1CCN(C(c2c(CC)nns2)=O)C2C1C2 15659,CC(C)C(C(=O)NCC1(C(=O)NC2CCOC2(C)C)CCCO1)NC=O 15660,c1(OC)cc(C(=O)NC(C)CCCCNC(C2CCC3(CC3)C2)=O)cc(OC)n1 15661,C#CCC(C(=O)NC(CO)CC(C)C)NC(c1cnc(CC)nc1)=O 15662,c12nccc(c1F)CN2C.C1(Cc2ccccc2)CCCN(CCO)C1 15663,C#Cc1ccc(C(=O)N(CC(=O)NC(C)Cc2ccco2)C(C)C)o1 15664,C=C(F)C1(CC(=O)NCC(C)NC(=O)CCCC(=O)OCC)CCOCC1 15665,n1(CC(=O)NC2CC(N(C(C)=O)C)C2)cc(C(F)(F)F)cn1 15666,C=CCC(CC(=O)NC(C)CCOC)NC(=O)Cn1nc(C)oc1=O 15667,C1(CNC(C(C)(C)OC(C)=O)=O)CN(C(=O)CN2CCS(=O)(=O)CC2)CCCO1 15668,c1(C(=O)NCCNC(c2c(C)nsc2)=O)c(Cl)cc(F)cc1Br 15669,c1(CN2C(C(=O)NCCCC)CC3(CC3)C2)c(F)cc(Br)cc1Br 15670,C1(C)(C(=O)NC(C(CO)NC(c2cc(CSC)c(C)s2)=O)C)CCC(=O)N(C)C1 15671,CC(C)C(CCO)N=c1ccnc(NC2CNC(=O)C2)[nH]1 15672,C1(CNC(C2(C(=O)NC)CCC2)=O)CCN(C(=O)C(C)O)CC1 15673,C(CCCCC(=O)NC1(C)CC(C(N2CC(O)C(O)C2CO)=O)C1)OCC 15674,C1(C(=O)NCC(C)(C)OCCNC(CCC(=O)OCC)=O)CC12CCCOC2 15675,N1(C(c2c(SC)csc2)=O)CC(NC(=O)Cc2cc(=O)n(CC(C)C)[nH]2)C(O)C1 15676,c1(OC)cc(=NC(=O)CC2CCC(NC(c3n[nH]cc3C)=O)CC2)[nH]n1C 15677,N1(C(C(CC)COC)=O)CCCC12CCN(C(c1cnc(O)n(C)c1=O)=O)C2 15678,c1(C(N)=O)ccc(NCC2CCN(C(C3CCOCC3(C)C)=O)C2)c([N+](=O)[O-])c1 15679,CC(CNC(=O)C1=NNC(=O)C1)C(F)C(=O)NCCCc1cnn[nH]1 15680,C(=O)(C(CCCCCN)C(C)C)N(C12CC3CC(C1)CC(F)(C3)C2)CC 15681,C1(c2onc(C(c3ccccc3F)CF)n2)CC(C(F)(F)F)C(O)C1 15682,N1(C(C2C3(CCC3)C23CCC3)C(=O)NCSc2ccccc2)CCC(F)(F)C(O)C1 15683,c1(C(N(C)CC2COCCN2C(c2n[nH]c(=N)[nH]2)=O)=O)cc2cnccc2[nH]1 15684,C(=O)(CCC1=NNC(=O)CC1)NC1(CNC(c2c(SC)cn(C)n2)=O)CC1 15685,C(CC(F)F)(C(=O)NC1C(O)CC1O)N(C)C(C1CCC1)=O 15686,CCC(CNC(C1CC(=O)CN1C(=O)CSCC(N)=O)=O)(CC)CO 15687,C1(C)(C(N(CC(CNC(C(C=C)O)=O)(C)C)C)=O)CCC2CC2C1 15688,C12(C(N3CC4C(NC(c5c(CC)scc5)=O)C4C3)=O)CCC(CC1)C(C)O2 15689,Cc1cc(=NCc2csc(Br)n2)[nH]c(=NCc2nc(C(C)(C)C)n[nH]2)[nH]1 15690,Cc1ccc(CC(=O)NC2CN(C(=O)CCc3cccn3C)CC2C)c(Cl)c1 15691,c1(C(=O)NCC2C(Cn3cc(COC(C)C)nn3)C2(F)F)cccc2c[nH]nc12 15692,Cc1ncsc1C=CC(=O)N(CCC(C)NC(=O)CS(=O)(=O)NC1CC1)C 15693,C1(CNC(C(CC)N(CC)CC)=O)CCN(C(c2cncc(OC)c2)=O)CC1 15694,c1(C(=O)NC2C(OC)CN(C(c3cnn(C(F)F)c3)=O)C2)ccc2cc[nH]c2n1 15695,C1(C(=O)NC2CC2NC(=O)Cc2ccn(C)n2)(COC)CCCO1 15696,C1(c2ccc(CC)o2)COCCN1C(C(=O)NCc1ccccc1)c1ccon1 15697,c1(CNC2CCC(C(=O)Nc3c(OC)nnc(Cl)c3)CC2)c(F)ccc(F)c1O 15698,C1(NC(CNC(C)=O)=O)C2CN(C(C3CCCN3Cc3nnn(C)n3)=O)CC12 15699,c1(OC)c[nH]c(C(=O)NC(C)CCCCNC(=O)C(F)n2cccn2)cc1=O 15700,N1(C(C2CCCC2NCC2CCCC3CCCCC23)=O)CCOc2ccccc21 15701,N1(C(Cc2nc(C)sc2)=O)CC(NC(c2ccsc2Br)=O)C2CC2C1 15702,C1(NC(=O)COC2CCN(C(C34CCC(CC3O)C4)=O)C2)CC2C=CC1CC2 15703,C1(NC(=O)CCc2ccc[nH]2)CCC(NC(C2(C(F)(F)F)CCC2)=O)C1 15704,N1(C(C2(CC)CCOCC2)=O)CC2CC(NC(c3cn(C)cn3)=O)CC2C1 15705,Cc1ccc2ncc(C(N3CCC4CCN(C(C5(F)CC5)=O)CC4C3)=O)cc2c1 15706,c1(C(N2CC(C)(NC(c3cncc(CC)c3)=O)C2)=O)c(C)cc(F)cc1Br 15707,CC1CN(Cc2ccnn2C)CCC1OC(C1CCCN(C(C)(C)C)C1)=O 15708,N1(C(C(C2(O)CN(C(c3cccnc3O)=O)C2)F)=O)CC2C(C1)C2(F)F 15709,N1(C(C2(C)CC2)=O)CC(C)CN(C(c2ccc(C3CC3)cn2)=O)C(C)C1 15710,N1(C(C2CC(CC)C2)=O)C(C(=O)NOC(C)(C)C)CCC1C1CC1 15711,C#CCC(O)C(=O)NC(C(=O)NC1CC(CC(N)=O)C1)C1CCOC1 15712,C1(NC(C(F)=CC)=O)CC2CCC1CN(C(c1cc(C(F)(F)F)ccc1C)=O)C2 15713,c1(C(=O)NC2C(C)(CNC(C3C(=C)C3)=O)CCC2)c(S(C)(=O)=O)cnn1C 15714,CS(=O)(=O)CC(=O)NC(C(=O)N1CC(CC(F)F)C1)C1CC1 15715,CC(CCCCCO)NC(c1nnnn1CCC1CC1)C1(C)CCCC1 15716,c1(NC(C2CC(CCNC(C3C(OC)CC3)=O)C2)=O)cnn(CC2CC2)c1 15717,Cc1cnccc1C(=O)NC(CNC(=O)C(C)NC(c1cccs1)=O)C1CCC1 15718,Cc1cnccc1C(C)C(=O)NCC(C)(C)CN(C)C(c1[nH]cnc1C)=O 15719,C1(NC(c2cccc(CC)n2)=O)CN(C(=O)C(C)n2cnnn2)CC1S(C)(=O)=O 15720,N1(C(C2(CC)CCCC2)=O)CC(C(N2CCCC(C(C)C)C2)=O)C(F)(F)C1 15721,CN1CC=C(CC(=O)NC2(CF)CN(C(c3cnc(S)[nH]3)=O)C2)CC1 15722,C(=O)(CCCCC(=O)OC)NCC1CCC(N(C(C(CCOC)OC)=O)C)CC1 15723,CCCCC(COC)NC(C1(CF)CCN(C(=O)C=CC(F)(F)F)C1)=O 15724,C1(C(=O)NCc2cn(CC#C)nc2)COCCN(C(=O)Cc2scnc2C)C1 15725,c1(C(=O)NCC2N(C(=O)C3=CCCSC3)CCC(C)C2)cnc2ccoc2c1 15726,C1(C(N(C2CC(OCC)C2)C)=O)CCCC1CNC(C1CCOC1CC)=O 15727,N1(C(=O)CCCc2cnn[nH]2)CCN(C(C2CC3(CCC3)C2)=O)C(CO)C1 15728,N1(C(C2(OC)CCCOC2)=O)CCC=C(CNC(=O)C(C)C(C)C)C1 15729,C1(CN(C(c2cc(CNC(CCCC)=O)on2)=O)C)CCCCCC1 15730,C1(CC)CN(C(c2cc(CC(C)C)c[nH]2)=O)CCN1C(=O)C=C1CCN(C)C1 15731,Cc1nnc2n1CCCC2C(=O)NC1CN(C(=O)C(c2ccnn2C)C)C1 15732,c1(C(=O)NC2C3CN(C(c4cnc(C)nc4)=O)C(C3)C2)ccc2c(c1)CCC=C2 15733,c1(CC(=O)NCC(C(C)C)NC(C(n2c(C)ccn2)C)=O)cnn2ccccc12 15734,C(=O)(C(C)(C)C)NCC(n1cc(C2CCCC2O)nn1)C.C1(=O)CN1 15735,Cc1cc(C(=O)NC2(C(=O)NCc3nccn3C(C)C)CSC2)cnn1 15736,Cc1nn(C)c(C(=O)NC2(C#N)CCN(C(c3cnnn3C)=O)C2)c1F 15737,C(=O)(CCC(CF)CF)N1CC2C(NC(c3n[nH]c(C)c3O)=O)(CC2)C1 15738,c1(CCC)nc(C)c(C(=O)NCCNc2ncc(C(=O)OC)cn2)s1 15739,c1(CC(N2CC(CC(C)(C)C)C(NC(C3CC34CC4)=O)C2)=O)ccc(Cl)cc1F 15740,c1(C2(C(=O)NC3(CC4CC4)CC3)CC2)cccc(C#N)c1.CC1CNC(=O)C1 15741,C(CCN=c1[nH]c(=NCC(C)C2CCC2)[nH]c2c(F)cccc12)N(CCOC)C 15742,C(CCCC1CC1C)NC(C1(NC(CC2(SCC)CC2)=O)CC1)=O 15743,CC1CC(C(=O)NCC(O)C(=O)NC(c2nn[nH]n2)C2CC2)CN1C 15744,c1(C(=O)NCC2(F)CCC(NC(CCC(C)OCC)=O)C2)cnc(C)nc1CC 15745,N1(C(CCC2C(C)(C)C2)=O)CC2CCCC2(CNC(=O)COC(=O)CO)C1 15746,c1(CC(N2CC(N(C(=O)C=Cc3cnc[nH]3)C)C2)=O)ccc([N+](=O)[O-])cc1 15747,C12(CC(=O)NCC3CCCCC3N3CCOCC3)COC(CF)(C1)C2 15748,C1(NC(CC(c2cccs2)NC(C)=O)=O)CCCN(C(c2cc[nH]c(=N)c2)=O)C1C 15749,c1(C(N(C(C)CNC(c2c[nH]c(C#N)c2)=O)C)=O)ccc([N+](=O)[O-])s1 15750,C(=O)(C(O)C(F)F)N1CCC(N(C(COCCOCC)=O)CC)C1 15751,c1(C(=O)NC2C(CNC(c3ccn(CC)n3)=O)CC2)cc(Cl)cc2c1NCCC2 15752,N1(C(C2(CNC(CN(C(COC)=O)C)=O)CCCCC2)=O)CC(F)(F)CCC1C 15753,C1(C(=O)NC(c2nc[nH]n2)CC)CSCCN1C(=O)CCC1CCCC1 15754,N1(C(c2c(C)cco2)=O)CC2(CC(NC(=O)C(F)C3CCC3)CO2)C1 15755,C1(C(N2C(C)(CNC(CSCCC)=O)CCC2)=O)COCC(C)(C)O1 15756,c1(C(=O)NC(C(CC)CC)C)n[nH]c2c1CN(C(C1(F)CC=CCC1)=O)C2 15757,N1(C(c2cnc(CNC(C3(C)CCCC3)=O)nc2)=O)CC2CCCC(O)C2C1 15758,Cc1cnc(Br)c(NC(C2CC23CN(Cc2nc(Br)cs2)C3)=O)c1 15759,N1(C(C2(SCC)CC2)=O)CC(NC(=O)C=C(C)c2ccsc2)C(O)C1 15760,C12(C(N(CC(O)CNC(C3C=CCC3)=O)C)=O)C3CC(CC13)C2(F)F 15761,C1(C(=O)NC2CC(N(C(C(C)CC3CC3)=O)C)C2)OCCCC1(C)C 15762,C1(O)(CNC(c2nn(C)c(F)c2)=O)CCN(C(=O)CC2CCCC(=O)N2)CC1 15763,N1(C(CCC(=C)Cl)=O)CC(NC(c2cnn(-c3ccccc3)c2F)=O)CCC1C 15764,c1(NCCC(C)OC)[nH]c(=NCC2OCc3cc(Cl)ccc32)nc2c1cnn2C 15765,c1(OC)cccnc1C(=O)NCC1CCC1NC(=O)CC(C)CF 15766,N1(S(C2CC(OC)C2)(=O)=O)c2ccccc2C(C)(C)C1C 15767,C(C(C)(C)NC(=O)CCC1(C)CC1)N(C(=O)CC1CCCO1)C.C1(=O)C(C)N1 15768,N1(C(c2n(C)nnc2)=O)CCOC(C(=O)NC2COC3(CCC3)C2)CC1 15769,N1(C(C2N(C=O)CCC2)=O)CC2(CNC(C3CCCS3)=O)CC(F)(C1)C2 15770,c1(C(=O)NC2(CNC(C3CC(C)(CC)C3)=O)CCOC2)cncc2c1CCC2 15771,c1(CCOCCNC(c2n(CCSC)nnn2)C2CC2)cccc(Cl)c1C 15772,CC1CCCC1(C(=O)Nc1ccccc1)NC(=O)C(c1cncnc1)C 15773,CCC(CC)(CCNC(C1(F)CCOC1)=O)NC(c1ccc(C)c(Cl)c1)=O 15774,C1(C(=O)NC(C2CCCO2)(C)C)COCCN1C(=O)C=CC1CCOCC1 15775,Cc1[nH]nc2c1CCC(C(N1CCC(C)(CNC(c3c(Cl)n[nH]c3C)=O)C1)=O)C2 15776,Cc1cc(F)c(F)cc1C(=O)NC1CN(Cc2ccc(F)c(O)c2)CC1F 15777,Cc1cc[nH]c1NC(C1CC(CC(=O)NC2(c3ccnn3C)CC2)C1)=O 15778,C1(C(N2CCCC(OCCC)C2)=O)CCN(C(=O)CCC2CCC(=O)C2)C(C)C1 15779,CCCCCCCCC(=O)NCC(C)(CC(C)C)NC(C1CC1C(N)=O)=O 15780,N1(C(C(C2CC2)SC)=O)CCN(C(c2cccc(F)c2O)=O)CC(O)C1 15781,c1(C(=O)NCC(CO)NC(=O)C(C2CCCC2)C2CCC2)ccc2c[nH]nc2c1 15782,C1(NC(Cc2c(C)noc2)=O)CCN(C(c2ccc(C3CC3)cc2)=O)CC1 15783,N1(C(CCc2cn(C)nc2)=O)CCN(C(C2COC(C)(C)CO2)=O)CC(O)C1 15784,c1(Nc2cncc(CNC(C3C=CC(CC)C3)=O)c2)ccc(C)c(C(F)(F)F)c1 15785,c1(C(=O)NCC2(NC(c3c(C#C)c[nH]n3)=O)CCCCC2)cc(C)ccc1O 15786,CCC(CC(=O)NCC(C)(C)NC(=O)CCCNC(c1ccsc1)=O)C(C)(C)C 15787,Nc1cnc(C(F)(F)F)cc1C(N1CCC(F)(CNC(C2CC(F)C2)=O)C1)=O 15788,S(=O)(=O)(c1cncc(Br)c1)N(CC)Cc1cccc(C2CC2)c1F 15789,C1(O)(CCNC(c2cn(C3CCOCC3)nn2)=O)CCN(C(=O)C=C2CCC2)C1 15790,C1(C(=O)NCC(C)C#N)CC(N=[N+]=[N-])CN1C(=O)CC(C)(C)C#N 15791,c1(C(=O)NC(CO)C(O)C2CCCCC2)cnn2ncccc12 15792,c1(OC)cc(CCC(=O)NC23CC(NC(C4CCCO4)=O)(C2)C3)ccc1O 15793,c1(OCC)cccc(C(=O)NC2CCC(CCNC(C3(OC)CC3)=O)C2)c1 15794,CC(C)C(C)C(C)CC(=O)N1CC2(CC2)CC1CNC(c1cccc(F)n1)=O 15795,C12(NC(c3ncn(C)n3)=O)CC1CN(C(c1cncc(C3CC3)c1)=O)C2 15796,C1(c2cn(CCOCCN(C(c3nnc(Br)s3)=O)CCO)nn2)CCCCCC1 15797,C1(C(C(=O)NC2CCC2)N(C2CCCOC2)C)CCC2CC2C1 15798,C(=O)(C1CCCc2ncnn21)NC(C(C)CSc1ccc(S(N)(=O)=O)cc1)=O 15799,N1(CCC)CC(C(=O)NCCC2(C)CCN(C(c3cncnc3C)=O)C2)CC1=O 15800,CC(C)CC(C)(O)C(=O)NCC12CCC(CC1)N(C(C1CCSCC1)=O)C2 15801,C(CC(F)=C(F)F)NC(C12CC(NC(=O)C=Cc3cc[nH]c3)(C1)C2)=O 15802,c1(C(=O)NCCC(C(C)C)C)cccc2c(Cl)cccc12 15803,c1(OC)nsc(CNC(c2nnc(C(F)F)o2)C(C)C)c1Br 15804,C1(CC=C)(NC(c2cnccc2C)=O)CCCN(C(C2CC(OC)C2)=O)C1 15805,N1(C(c2ccn(CCC)n2)=O)CC2CN(C(=O)Cc3cc(O)nnc3O)CCC12 15806,N1(C(C(C)NC(C2CCC2)=O)=O)CCCCC1CN(C)C(C1(F)CCOCC1)=O 15807,c1(NC(N2CCN3CC(F)(F)CC3C2)=O)cc2c(cc1Br)OCCO2 15808,Cc1ccc(C(C)CC(=O)NC23CC(NC(c4cncc(N)n4)=O)(C2)C3)cc1 15809,C1(C(=O)NC2C(NC(c3c(C)nn[nH]3)=O)CC2)CCCC2(CC2)C1 15810,C1(C(=O)NC2CC(CC(=O)NCC3(OC)CCOC3)C2)CC2CC1CC2O 15811,c1(C(=O)NCC(N2CC3CC2CC3CNC2CC2)=O)c[nH]c2cc(F)c(F)cc12 15812,c1(C(C)(C)C)ccc(C(=O)NC2CC2CNC(=O)C=Cc2cncs2)nc1 15813,c1(C(=O)OC(c2ccccc2Cl)C(=O)OCC)ncc(Br)cc1C1CC1 15814,c1(NC(=O)NC2C(O)CCC(C)C2)ccc([N+](=O)[O-])cc1I 15815,c1(NC(C2C3CN(C(C(C)Cc4ccccn4)=O)C2C3)=O)cc(Cl)nnc1Cl 15816,C1(CC(=O)NCC(C(C)C)(C)NC(C2C(F)(F)C23CC3)=O)CCCCCCC1 15817,C(=O)(C1=CNS(=O)(=O)N=C1C)NC1CN(C(C2CCN(C(CC)=O)C2)=O)CC1C 15818,c12ccc(cc1)N(C=O)C2c1cncnc1.c1(C2CC(=O)NC2)ccc(Br)cc1 15819,N1(C(C2OCC(C)C2)=O)CCOCC(CNC(=O)CC2NC(=O)NC2=O)C1 15820,C(=O)(C1=CNC2=NCCC2=C1)N1CC(O)(CNC(=O)CC2CCCCCO2)C1 15821,C1(NC(c2c(OCC)nc(Cl)cc2)=O)CC2CN(C(=O)C(C)(C)O)CC2C1 15822,CC(c1ccccc1Cl)=CC(=O)NC(C1(O)CN(C(C2(C)CC=CCO2)=O)C1)C 15823,c1(CC(=O)N(CC(CC)NC(c2cc(C)c[nH]2)=O)CC)cnc(C(C)C)[nH]1 15824,CC(C)CC(C(=O)NCC(C)(C)CCNC(=O)CC1CCCN1C)C(C)C 15825,C1(CC(=O)NCC=CCNC(C2CC3OC(=O)OC3C2)=O)CCc2sccc2C1=O 15826,C(CCS(=O)(=O)c1ccccc1)NC(=NCCCSCC)NC1CCS(=O)(=O)C1.C=CC 15827,c1(C(N(C2CC(NC(CN(CC)CC)=O)C2)C)=O)cnn2c1CCCC2 15828,N1(C(C(C)=CC)=O)CCC(NC(=O)CC(O)c2ccccc2)C1(C)C 15829,c1(C(N2CCC(NC(C(CCOC)C)=O)(CO)CC2)=O)cc([N+](=O)[O-])ccc1C 15830,N1(C(C=CC)=O)CC2ON=C(CNC(=O)C(C)=C3CC3)C2C1 15831,N1(C(CCCN(C)C)=O)CCN(C(=O)CCCC2CCOCC2)C(C2CC2)C1 15832,n1(CC)nc(C2CC2)cc1C(=O)NC1CN(C(=O)COC(C)=O)CC1SC 15833,C1(S(N)(=O)=O)(C(=O)NCCNC(C(c2ccc(Cl)cc2)(C)N(C)C)=O)CCCC1 15834,C1(C(N(C2CN(C(c3n[nH]c(C)c3O)=O)CC23CC3)C)=O)CCc2cnnn2C1 15835,CC1(NC(C2CC(NC(=O)C=C3CCC3)C2)=O)CCC(O)CC1 15836,C=CCC(C(=O)NCCCOC1CCCCCC1)C(C)C 15837,c1(C(=O)NC2CC(C)(NC(c3cnc(C4CC4)s3)=O)C2)ccc(C(F)(F)F)cc1 15838,C(=O)(C1COc2ccc(F)cc21)N1CCC(NC(C2(C(F)(F)F)CC(=C)C2)=O)C1 15839,c1(C(=O)NC2(CC=C)CN(C(c3cnc(Cl)s3)=O)C2)cnn2cnnc2c1 15840,c1(SC)c(C(=O)NC2CCCCC2NC(c2nc(C3CC3)oc2C)=O)cnn1C 15841,c1(CSCC)ccc(C(=O)NC(C)CC2CN(C(=O)C(F)CC)C2)cc1 15842,c1(C(N2CC3CC2CO3)=O)cc2n(n1)CCCN(Cc1cc(F)c(Cl)c(F)c1)C2 15843,N1(C(CC2CC(=O)C2)=O)CCC(C2(CNC(C3CCCSS3)=O)CCOCC2)CC1 15844,c1(CN2CCN(CC(=O)Nc3cnc[nH]3)C(=O)C2)cc(F)c(O)cc1F 15845,C=C(C)C1OCCC1C(N1CCCCC1CNCc1cc(OC)cc(OC)c1)=O 15846,c1(OC)ccc(OC)c(CCC(=O)NCC(C2CCC2)NC(=O)CC=C(C)C)c1 15847,c1(C(N2CCN(C(CCC3N(C(C)=O)CCC3)=O)CC2)=O)ccc(F)c(Br)c1F 15848,CC(C)C(CNC(c1cn(CC2CC(=O)C2)nn1)=O)NC(C1CC12CCC2)=O 15849,c1(C(N2C(CN(C)C(C3CCC(C)(C)O3)=O)CCCC2)=O)ccc2ncsc2c1 15850,C1(NC(=O)CCC2CC2)CCc2onc(C(=O)NCC(F)F)c2C1 15851,N(C(=NCCc1ccnn1C)NCC(C)(C)C)C1CCN(C(=O)OC)CC1 15852,N1(CC(=O)N(CC(C)(C2CC2)NC(=O)C#CC(=O)N(C)C)C)CCC(CO)CC1 15853,C1(NC(C=CC)=O)CCN(C(=O)CCOc2ccccc2C(N)=O)C(C)C1 15854,c1(C(N2CCC(C(CNC(C(CC)NC(C)=O)=O)C)CC2)=O)c[nH]c(=N)cc1C 15855,C(c1nc(C)co1)=CC(N1CC(NC(CC(c2ccccc2F)OC)=O)C1)=O 15856,C12(CNC(c3n(C)ccc3)=O)CCCC1CCN2C(c1csc(CO)n1)=O 15857,CC(CN=c1nc(N2CCOC(c3ccccn3)C2)c2c([nH]1)COC2)N(C)C 15858,c1(OC)cc(C)cnc1C(N1CC(CNC(c2cc(C)co2)=O)C(C)(C)C1)=O 15859,C1(NC(C(CN(C)C)O)=O)C2CCN(C(=O)CCSc3nnnn3C)C12 15860,CCC(C(=O)N1CCCC1CC(=O)NC(C)(C)C#CC)NC(N)=O 15861,C(c1ccoc1)=CCOCC(N1C(CC(=O)NC(C2CCOC2)C)CC1)=O 15862,N1(C(CN2C(C)CCC2)=O)CC2CC1CCC2NC(c1ccc(F)c(CO)c1)=O 15863,Cc1cccc(OCCC(N2CC(NC(=O)Cc3occc3C)C(C)C2)=O)c1C 15864,c1(C(=O)NC2C(NC(C(CC)N(C)C)=O)CCOC2)cccc2[nH]cc(C#N)c12 15865,C1(C(N(CCNC(C)=O)C)=O)CC2CC1CC2NC(c1cncc(O)c1)=O 15866,Cc1cc(C(=O)NCC2CCN2Cc2ccsc2Cl)ccc1[N+](=O)[O-] 15867,N1(C(C2CCC(=O)N2)=O)CCCCC1CNC(C1CCC(O)CC1)=O 15868,c1(C(N(C(CC(C)C)C(=O)Nc2cnn(C)c2)C)=O)ccn2ccccc12 15869,C#CCCCC(C)C(=O)N1C(CNC(=O)Cn2ccccc2=O)CC2CCCC12 15870,C(=O)(C(C)CNC(C1CCSCC1)=O)NC(c1ncco1)C 15871,C#CC1(c2ccccc2)COCCN1C(=O)NCCc1cn(CC)cn1 15872,C=CCC(F)(F)C(=O)N1CCN(C(C2CC23CC(OCC)C3)=O)C(CF)C1 15873,N1(C(c2scc(COC)c2)=O)CC(C)(CNC(=O)CCCC(C)(C)C)CC1(C)C 15874,N1(Cc2ccc(C#N)cc2)CCC2CN(C(c3csc(Br)c3)=O)CC2C1 15875,c1(OC)cc(Br)ccc1C(CO)NC(C1C(CN)C1(C)C)=O 15876,C=C(C)CCC(=O)NCC1(O)CC(CNC(=O)CNS(=O)(=O)CCCOC)C1 15877,N1(c2nnc(C)o2)CCC2(CCC(NC(c3cc4c[nH]nc4cc3C)=O)CC2)C1 15878,CC1(F)COCCN(C(=O)Nc2cccc(C3CC(F)(F)C3)c2)C1 15879,C=C(C)CN=c1[nH]c(=NCC2(CS(C)(=O)=O)CC2)c2ccccc2[nH]1 15880,N1(Cc2n(CCCC)nnn2)CCCC2CN(C)CCC12 15881,c1(CC(N2CCN(C(c3cc(N)c(F)cc3)=O)CC2)=O)cnc2c(=O)[nH]ccn12 15882,CCCCCCC(=O)N1CCCC(CCC(=O)N(C2CCCNC2=O)CC)C1 15883,Cc1ccc(C)c(C(=O)NC2C=CC(CC(N3CCC4CC34C)=O)C2)n1 15884,N1(C(CC(CC)OC)=O)CCc2nc[nH]c2C12CCN(C(=O)C=CI)C2 15885,c1(C(=O)NC2C(CNC(COC)=O)C2)cc2ccccc2nc1C(F)F 15886,N1(NC)CCC2(CCCC2)CC1.Cc1nn(C2CC2)cc1-c1ccc(C)cc1 15887,c1(C(N2CC3C(C(N(C(C)C(N)=O)C)=O)(C3)C2)=O)c(O)cccc1F 15888,C1(N(C)C)(CNC(C2OCCC2NC(C2C=CCC2)=O)=O)CCOCC1 15889,C1(C(=O)NCCN2CCC(C)(C)C2)CCC(C)(C)N(C(=O)C=C2CC2)C1 15890,C1(C(C)C)CCN(C(C2(C)CN(C(=O)CCOC3COC3)C2)=O)CC1 15891,C1(C(=O)NCCC2N(C(Cc3nnc(C)s3)=O)CCCC2)CC2CCCCN2C1 15892,C1(NC(CCCc2[nH]c(=N)sc2)=O)CN(C(c2cccc(=O)o2)=O)CC2CC12 15893,c1(OCC)cc(C(=O)NC(C)CC2CN(C(=O)CSSC)C2)[nH]n1 15894,C(=O)(CC(O)CCCCC)N1C(C#C)CN(C(=O)CSC(C)(C)C)CC1 15895,N1(C(CCCC2(NC(C(COC)C)=O)CCC2)=O)CC2(C1)CN(C)C2 15896,c1(OC)ccccc1C1(NC(N2CC(n3c(O)nnc3O)C2)=O)CCC1 15897,C1(C(N2CCC(CNC(CCN(c3ccncc3)C)=O)C2)=O)CCC2(CC2)C1 15898,CCCCC(=O)C(=O)N1CCCC1C(C)NC(=O)CCOc1ccc(Cl)cc1Cl 15899,C(C1CC1)(C1CC1)=CC(=O)NC1CC(NC(C2CSCC2c2ccccc2)=O)C1 15900,C(=O)(CS(=O)(=O)C(C)(C)C)N1CCC(OC)(CNC(C2CCC(CO)CC2)=O)C1 15901,N1(C(c2cccc(SC)c2)=O)CC2CCC1CN2C(=O)C(C)(C)F 15902,c1(CC(N2CCC(C)(c3cn(CCCO)nn3)C2)=O)c[nH]c2ncc(Br)cc12 15903,C(=O)(C(C)C(F)(F)F)N(C(C)C)CCN(C(=O)C(O)Cc1ccc(Cl)cc1)C 15904,C(=O)(C(F)(CNC(=O)CCc1cnco1)C(C)C)NC(C)Cc1cccs1 15905,c1(C(=O)NCCC2CCN(C(C(C)OCCOC)=O)CC2)nccc2n[nH]cc12 15906,C(CCCC(=O)NCC1CCC(NC(=O)CC2CCCN2C)CC1)N(C(C)C)C 15907,C1(c2cccc(F)c2)(NC(CCOCCC)=O)CCN(C(=O)C=NOC)C1 15908,C(c1cccc(O)c1)=CC(=O)NCC1CN(C(c2cccc(C)n2)=O)CC1C 15909,C1(NC(c2c(CC)noc2)=O)CCC12CN(C(c1cccc(F)c1OC)=O)C2 15910,O=C1CCC(CC(N2CCC(O)(C(F)F)C2)=O)CN1 15911,N1(C(c2noc(CC)c2C)=O)CC(C)CN(C(=O)C2=NNC(C(F)(F)F)C2)C(C)C1 15912,C1(C(=O)NC2(CC(=O)NCc3ccccc3Cl)CCC2)CCC(F)(F)CC1 15913,c1(C(N2CCC(CNC(C(CCC)OC)=O)C23CC3)=O)cc2ccncc2[nH]1 15914,N1(C(CC(C)(F)F)=O)CC(O)C(O)C1CNC(=O)CC1CC(O)C12CCC2 15915,C1(C(=O)OC(CC(=O)OCC)CC#N)CC2(CCCCC2)C1 15916,C#CCC(C)(CC)C(=O)NCCCC(=O)NC1CC12CCCC2 15917,C(CCCCC(=O)NC1(C2CCCCN2C(=O)C(C)n2cccn2)CC1)OCC 15918,Cc1cnccc1CN(C)C(c1cc(C2CC2)nn1C(C)(C)C)=O 15919,C1(NC(=O)CCc2ccoc2)CC2CC1N(C(C1(c3ccc(F)cn3)CC1)=O)C2 15920,C1(CN(C2CCCC2)CC(=O)NCC(F)F)CCC(C(F)F)CC1 15921,N1(c2n(CC(=C)C)c(Cc3cccnc3)nn2)CCCc2ccccc2C1 15922,C1(C2(O)CN(C(C3(Cl)CC3(F)F)=O)C2)(CNC(C(F)=C(C)C)=O)CC1 15923,c1(C(=O)NCCCN(C(c2c(C)[nH]c(C)c2C)=O)CC)cccc(C(N)=O)c1C 15924,C(C)(CCCCN=c1nc2c(cnn2C)c(NCC(C(C)C)C(C)C)[nH]1)OC 15925,Cc1csc2ncnc(N3CCCCC(CNC(=O)CCc4cscn4)C3)c12 15926,c1(CCOC)n[nH]c(=NCCCNC(C2CCCC2OCc2cccc(Cl)c2)=O)s1 15927,c1(-c2cc(C(=O)OC)sc2)ccc2c(c1)CCN(c1cc3ncnn3cn1)C2 15928,c1(N2CC(C(C)NC(c3cccn3CCC)=O)OCC2)ncnc(Cl)c1C#N 15929,O=C(C1=NOC(CNC(C2(O)CCSC2)=O)C1)NCCC12CC(CO1)C2 15930,c1(CC(N2CC(CCNC(C)=O)C2)=O)c(N)nc(C)nc1O 15931,C(C(C)CC(F)(F)F)OCC.c12cccc(c1)N2C(=O)OC(C)(C)C 15932,Cc1csc2ncc(C(=O)NC3CCCN(C(C4CC5(C4)CC(O)C5)=O)C3)n12 15933,N1(C(c2cc(O)cs2)=O)CC2CC(C1)N(C(=O)CC1CCCC3(CCC3)O1)C2 15934,C1(n2cc(CCNC(C3(C)C(C)C3)=O)nn2)CCCC=C1Br 15935,C1(N(C(=O)Nc2ccccc2)C2CC2)CCN(C(c2ncccn2)=O)C(C2CC2)C1 15936,c1(C(=O)NCC2(CNC(C=Cc3cc(C)no3)=O)CC2)ccccc1S(C)(=O)=O 15937,C1(NC(c2n(CC)ncc2)=O)CC2CCC(C1)N2C(c1nonc1N)=O 15938,N1(C(C(=CC2CCCC2)C)=O)CCCC(NC(=O)C(C)(C)CC2CCC2)C1 15939,Cc1cc(=NC(=O)C=CCC2(NC(c3cnn(CCF)c3)=O)CCC2)[nH]n1CO 15940,N1(C(c2n(CCC)ccc2)=O)CCC(CN(C(C2CNC(=O)O2)=O)CC)CC1 15941,Cc1cc(NC(C2CN(Cc3cccc(C#N)c3)CCO2)=O)cnc1F 15942,Cc1cc(CNC(=O)NCC2(Br)CCCCC2)nc(O)n1 15943,C1(C2CCN(C(C(=C(C)C3CC3)F)=O)C2)CCCCN1C(=O)CC1CCCOC1 15944,CC1CC(C)N(C(=O)C2CC2)CCN1C(c1nc2cc(Cl)ncc2s1)=O 15945,c1(C(=O)NCc2cc(C)cc(F)c2)ccc2c(c1)CCC2NC(=O)OC(C)(C)C 15946,c1(C(N2CC3CCN(C(CCOCC#C)=O)C3C2)=O)cnc2c(c1)CCOC2 15947,C1(NC(c2c(CC)cno2)=O)CN(C(=O)Cc2cscn2)CCC1O 15948,C12(C(N3C(CNC(c4nccc(C(C)(F)F)c4)=O)CCC3)=O)CCC(CC1)OC2 15949,C1(N(C)C(c2ccn(C)n2)=O)CC2CC1N(C(=O)C(CC1CC1)CC1CC1)C2 15950,n1(CCC)nc(CC2CCC2)nc1-c1nc(-c2ccncc2)ns1 15951,C1(NC(C(C2CCC(=O)N2)C)=O)CCN(C(=O)CCc2nc(=N)[nH][nH]2)CC1(C)C 15952,Cc1csnc1C(=O)NC(Cc1ccoc1)C(=O)NC(C)CCC1CC1 15953,c1(C(N2C(CNC(c3cc(Br)c[nH]3)=O)CC2)=O)ccc2cnoc2c1 15954,C(=O)(C(F)CCCC)NC(C1CCN(C(CCC=CC)=O)CC1)CO 15955,C1(NC(c2cc(CC)n(CCO)n2)=O)CN(C(c2cccc(N)n2)=O)CCC1O 15956,c1(C(=O)Nc2c(CC)nnn2C)ccc(C(=O)OC)c(Cl)c1 15957,Cn1ncc2c1CC(C(N1CCC(CCNC(c3cnc(O)o3)=O)CC1)=O)CC2 15958,c1(C(=O)NC2(C(=O)NC(C3COCC3C(F)(F)F)=O)CSC2)cc(C)c[nH]1 15959,C1(CNC(=O)NCc2cnc(Br)s2)CC(O)CN1C(=O)C(Cl)(Cl)Cl 15960,C(N=c1[nH]c(N(CCCN2C(=O)CCC2=O)C)nc2c1SCC2)C1OCC(C)C1 15961,c1(NC(C2CC(NC(C3(C)CCC3)=O)C2)=O)nc(Cl)c(Br)cc1[N+](=O)[O-] 15962,N1(C(C2C(C#N)CC2)=O)CCC(C(=O)NCC2CC23CC3(F)F)(CO)CC1 15963,N1(C(CCc2c(OC)ccc(F)c2)=O)CCCC2(NC(=O)C(=O)N(C)C)CCCC12 15964,c1(C(C(N2CCCC3CCCCC23)=O)(F)F)ccc([N+](=O)[O-])cc1 15965,C(C(O)C(=O)NCC1CC(NC(C2(CCN3CCOCC3)CC2)=O)C1)N(C)C 15966,Cc1ccc(SC(C)C(=O)NC2CCC(NC(C3CCC(CO)CC3)=O)C2)cc1 15967,C12(NC(C(C)N(C)C(c3c[nH]c(C#N)c3)=O)=O)CC1COC21CCC1 15968,N1(C(c2c(CCC)occ2)=O)CCC(C2CCN(C(=O)CCCCO)C2)C1 15969,C(=O)(C(CCC)S(N)(=O)=O)NC(CCC)CCCNC(=O)Cn1nc(C)nc1C 15970,C1(F)(C(=O)NCC(CNC(C2(CC3CCC3)CC2)=O)CO)CCCOC1 15971,Cc1ccc(SCCC(=O)NC2CN(C(=O)C#CC(C)C)CCC2F)c(C)c1 15972,Cc1nc(C(N2CC(NC(=O)COc3cccc(F)c3F)CC2C)=O)cc(O)n1 15973,C=CCC(C)(C(=O)N1CC(CO)C1)OC.c1(C(=O)NCC)occc1CC 15974,N1(C(C(CC)SC2CNC2)=O)CCC2(CC1)CN(Cc1cccc(C)c1)CCO2 15975,C1(NC(c2ccnc(C)n2)=O)COC2(C1)CN(C(c1cc(C(F)F)ncn1)=O)C2 15976,c1(NC(c2c(CCC)[nH]cc2)=O)ccc(NC(C2CC2[N+](=O)[O-])=O)c(C)c1 15977,N1(CCNC(=O)C(=O)NCC2CC2F)CCCOC1=O 15978,c1(C(N(CCCN(c2nc(COC)nc(O)c2)C)C)=O)ccc(F)c(C#N)c1 15979,Cc1cc(C(=O)NC2CC(NC(C3CCCN(CC(C)C)C3)=O)C2)ncc1C#N 15980,C1(C2(O)CN(C(=O)C=C3CCCCC3)C2)(CNC(C2(CC=C)COC2)=O)CC1 15981,c1(C(=O)NC(CC)CNC(C2(CF)CC2)=O)ccc2c(n1)NC(=O)CO2 15982,c1(C(=O)NC2CN(C(=O)CC3CCC(F)(F)C3)C2)cnc2cccnc2c1 15983,c1(C(=O)OC)ncnn1C1CCN(C(N2CC(c3ccccc3)C2C(C)C)=O)C1 15984,C#CCC(C)(C(=O)NC1(CC)CCOC1)NC(c1nc(C)ccc1C)=O 15985,N1(C(c2cn(CCCOC)nc2)=O)CCC(C)C(CNC(C23CC(CO2)C3)=O)C1 15986,C1(NC(C=CC(=O)OCC)=O)CCCC12CN(C(C1CN(S(N)(=O)=O)C1)=O)C2 15987,CON1CCC(C(=O)NC2CC(N(C(=O)CCC3CCCC(=O)N3)C)C2)CC1 15988,c1(N(C(=O)Nc2nc(CC(=O)O)cs2)CC)cccc(Oc2ccc(Cl)cc2)c1 15989,C1(C(=O)NC(c2ccco2)COC)CN(C(=O)Cn2nc(C)nc2C)CC1C 15990,C1(N(C)C(c2ccc(-n3cnnc3)cc2)=O)CN(C(=O)C(C)(F)F)CCC1O 15991,c1(C(=O)NCC(CC)NC(=O)CC2CCC(C)(C)CC2)csc2cncn12 15992,CCCCCCC(C(=O)NCCN(C(=O)C(CCC)C(=O)OC)C)N(C)C 15993,CC(CC(=O)NC1(C2CCN(c3nc(Cl)ncc3C3CC3)C2)CC1)C(F)(F)F 15994,CC1(F)CN(C(=O)CNS(C)(=O)=O)CCN(C(=O)CN2CCC(F)CC2)C1 15995,CN1CCCCC1C(=O)NC(CNC(c1ccc(OC2CC2)cc1)=O)CO 15996,C1(C(=O)NCCC(=C)CNC(C2C3CC4C(C3)C24)=O)CC2(CC(OC)C2)C1 15997,N1(C(C2C(CC(C)C)C2)=O)CC(NC(=O)C(=O)N(C)C)C2(CCOCC2)C1 15998,Cc1cc2c(C(N3CC4CC(NC(C5CCC(C)CC5)=O)C3C4)=O)nccn2n1 15999,C(CC1=CCCCC1)N(CC(CO)C1CC1)C(=O)Cc1ccc(Cl)cc1 16000,O=C1C=C(c2nc3c(s2)CC(C(=O)NCc2cc(F)ccc2Br)CC3)CCC1 16001,C1(C)(NC(C2C3CN(C(C(CCCC)C)=O)CC32)=O)CCCC(C)(C)C1 16002,C1(C(N(C2CCCC(NC(=O)COCCCF)C2)C)=O)Cc2cccnc2C1 16003,C12(C(=O)NCC(C(=O)OC)Cc3ccccc3OC)CCCC(C1)C(=O)NC2 16004,C1(NC(=O)NC2CN(C(CCC)C)C(=O)C2)CCOCC1(C)C 16005,Cc1nc2cc(F)ccc2cc1C(=O)NC(C)CNC(c1ccnn1C)=O 16006,S(=O)(=O)(c1ccc(NCCCC2CC2(Cl)Cl)cc1Br)NCc1cncc(OC)n1 16007,c1(C(N2C(C(N)=O)CCOCC2)C(=O)NCC2CC2)c[nH]c2ccc(Cl)cc12 16008,C1(C(N(CC(=O)N(C2CCCC2)CCO)C)=O)CCC(=O)O1 16009,CC1(C)CC(NC(=O)C(C)(C)CC#N)CN(C(c2cnc(C3CC3)o2)=O)C1 16010,C1(NC(CCOCCOC)=O)C(C)(C)C(NC(c2cc(F)n[nH]2)=O)C1(C)C 16011,N1(C(C2N(C)C(=O)CC2)=O)CC2(CC2)CC1CNC(=O)CCC(F)(F)F 16012,C(C#CC(F)(F)F)NC(C1CCCN1C(=O)CNC(=O)NC1CCCC1)=O 16013,N1(C(C2=CC(C)(CC)C2)=O)CCC2(CCN(C(c3cc(N)cc(O)n3)=O)CC2)C1 16014,C1(C(=O)OCC)CC(NC(=O)NCc2ccnn2CC(F)F)CCO1 16015,C(CCCCC(=O)N1CCOC(CNC(c2cc(C)cnc2C)=O)C1)OC 16016,Cc1cc(F)cc2[nH]c(C(N3CCC(CNC(c4ccc(F)cc4)=O)C3)=O)cc12 16017,C(=O)(C1=CCN(C(C2CC(=O)N(OC)C2)=O)C1)NC(CC)CCCO 16018,c1(C(=O)NC(C(=O)NC(C#C)Cc2ccco2)C2CC2)cc([N+](=O)[O-])c[nH]1 16019,C1(C(=O)NCC(C)CN(C(=O)C(F)CC2CCCCC2)C)CCC2(CC1)CC2 16020,c1(C(N(CCN(C(=O)CCc2cncnc2)CC)CC)=O)n[nH]cc1Br 16021,c1(C(=O)NCCC2CC(NC(CC=C)=O)C2)cn(-c2ccn(C)n2)cn1 16022,S(=O)(=O)(c1ccccc1)N(CC(N1C(CCCNC(C(C)SC)=O)CCC1)=O)C 16023,C1(C(=O)NC2C(NC(Cc3nc(C)c(C)o3)=O)CC2)C2CCC3C(C2)CC13 16024,C(=O)(C(CC(C)C)NC(=O)CC1CNC(=O)O1)N(C(CC)C1CC1)C 16025,N1(C(CC(C=C)(C)O)=O)CC2CCC(C1)C(NC(c1cnc(OC)c(C)n1)=O)C2 16026,C1(C)(C(N2CCC(CNC(C(CCCOC)C)=O)(OC)C2)=O)CCC2(CC1)CC2 16027,N=c1nc2c(c[nH]1)CCC21CCCN(C(=O)C(N2CCOCC2)C2CC2)C1 16028,N1(C(c2c(C)coc2)=O)CCCCCC(NC(=O)C(c2ccc(F)cc2F)C)C1 16029,C1(C(=O)NCC=C(C(=O)NC2(CC=C)CCCC2)C)CC12CCOC2 16030,CC(O)C(C)C(=O)NCC1CCCN1C(=O)Cc1csnn1 16031,C1(CC(C)C)CCN(C(=NCCc2ccccc2)NCC2CC2C(C)(F)F)C1 16032,C(=O)(CC(C)(O)C(F)(F)F)NCC(C)NC(CCC(=C)Cl)=O 16033,C1(NC(CSCC=C)=O)CC(C)(CNC(=O)C(C)CC2CC2)C1 16034,C1(C(N2C(C=C)CC2)=O)CCN(C(=O)CCC2CC(OC)C2)CC1(C)C 16035,N1(C(c2cc(C)nc(C)n2)C(=O)NC(CC)C)CCc2ccc(F)c(Br)c2C1 16036,N1(C(C23COCC2CN(Cc2cccnc2)C3)=O)CCC(C2CCOCC2)C1 16037,N1(C(c2cnc(C(C)=O)s2)=O)CCCC(C)(NC(C2C(F)(F)C23CCC3)=O)C1 16038,c1(C(N(c2c(C)cccc2Cl)C)=O)ccc(S(=O)(=O)Cc2nn[nH]n2)cc1 16039,c1(CC(=O)NC2CC2NC(=O)C=CC2CCOC2)cc(C2CC2)no1 16040,N1(C(C2N(C(C(C)C)=O)CCC2)=O)CCCCC(NC(=O)CCC(=O)N(C)C)C1 16041,c1(C(=O)NC2CC(NC(CC(=O)OC)=O)C(O)C2)ccc2ncncc2c1 16042,n1(C2CCCN(C)C2)ccc(=NC(=O)C(=O)N2CCC(N(C)C)CC2)[nH]1 16043,N=c1c(C(=O)Nc2cccc(Nc3ccccc3Cl)c2)c[nH]cc1Br 16044,c1(OCC(=O)NCCN(C(C(CCCC)C)=O)C)ccc2c(c1)CCCC2 16045,C(CC(C(=O)NCC1CCCC1(C)C)NC(c1cncc(C)n1)=O)=CC 16046,CCCC(C)(O)C(=O)NCC1CCCC1C(=O)NC1CN(C)CCC1O 16047,c1(C(=O)NCC2(COC)CCN(C(C3CC3(F)Cl)=O)C2)cc2ccccn2n1 16048,S(=O)(=O)(c1cccc(NC(N2CC(F)(CO)C2)=O)c1)N1CC(C)OC(C)C1 16049,C(=O)(CS(N)(=O)=O)N(CCCCCNC(C1(C)CC1Br)=O)C 16050,c1(C(N2CC(C)CC(NC(CC3(OC)CC3)=O)C2)=O)cc2n(n1)CCCO2 16051,C1(NC(c2c(SC)ccs2)=O)CCC(C)N(C(=O)C(F)C(C)C)C1 16052,C1(C(=O)N(C)CCNC(c2ccn(C(C)C)n2)=O)(CC)CCOC1 16053,CN1CC(C(=O)NC2CC(F)(CNC(=O)Cn3cnc(=N)[nH]3)C2)C(C(F)(F)F)C1 16054,C12(CNC(C(=O)N(C3CC(OC)C3(C)C)C)=O)CCC(O)C1CC2 16055,C1(CN(C(=O)CC2CCOC2)C)CN(C(=O)CCc2ccc[nH]2)CC12CC2 16056,CC1CCC(C(N)=O)CN1C(C1(C)CC1C(F)(F)F)=O 16057,C(c1cccc(F)c1)=CC(=O)NCC(C)(F)CNC(=O)CC12CCCC1C2 16058,C1(c2cccc(OC)c2)CCN(Cc2ccccc2N(C)C)C1(C)C 16059,CC(C)(C)C(C(=O)N1CCC(O)CC1C1CC1)Nc1cc(O)ccc1Cl 16060,N1(C(CC(CC)OC)=O)CC(C)(C)C(NC(c2cnc(Cl)s2)=O)C(C)(C)C1 16061,Cc1cccc(C(=O)NCCCCCNC(C2(C3CCCCO3)CC2)=O)c1O 16062,N(C(=NCc1c(Br)cncc1Br)N1CC(O)C(C)(C)C1)C(CC)C 16063,C1(NC(=O)Oc2ccc(Br)cc2Cl)CCCN(CCO)C1=O 16064,C1(CC)CCCN1C(=O)C(=O)NC1CCC1NC(C1(n2ccnc2)CCCC1)=O 16065,C(=O)(C(C)CC(F)F)N(C1CCN(C(c2ccc(SC)nc2)=O)CC1)CCC 16066,N1(C(CC2CC(=C)C2)=O)CCC2(CC1)CC(NC(=O)Cc1ccc(C)s1)CCO2 16067,Cc1cc(C(=O)NC(C2(C(=O)NCC3C4CCCCC34)CC2)C)sc1C 16068,CC1CC(NC(=O)C(C)C(=O)OC(C)(C)C)CCN1C(=O)CN1CCS(=O)CC1 16069,c1(C(N(CCC(C)NC(C(CN(CC)CC)F)=O)C)=O)cc(S(N)(=O)=O)sc1C 16070,N1(C(C(C(=O)OCC)CC)=O)CC2(CCN(C)CC2)C1 16071,C(CCC(=O)N(CCC(C)NC(=O)C(=O)NCC(F)F)C)=CC 16072,C1(NC(C(C)(C)n2cc(Cn3cc(Cl)cn3)nn2)=O)CC2CCCN2C1 16073,CC(C)C(C(=O)NC(C)CCN(C)C)NC(C1(CO)CC(C)(C)C1)=O 16074,CC1C(NC(=O)Cc2cnccc2Cl)CCCN1C(c1c[nH]c(C(F)(F)F)c1)=O 16075,c1(C(=O)NCC2CCN(C(C3CCCS3)=O)CC2)cccc2ncccc12 16076,C1(CNC(c2cnn(-c3ccncc3)c2)=O)C2CN(C(=O)CSC3CC3)CC12 16077,[N-]=[N+]=NC1CN(C(C2C3CC4C(C3)C24)=O)CC1NC(C1CC(O)CN1C(N)=O)=O 16078,N1(c2nnc(-c3c(CC)n[nH]c3)n2CC)CCC(S(=O)(=O)N2CCOCC2)C1 16079,C1(CNC(CS(CC)(=O)=O)=O)CN(C(=O)CC2(CSC)CC2)C2COCC2O1 16080,C=CCCN=C(NCCC(C)F)NC1CCOC(C(C)C)C1 16081,c1(OC)ccc(CC(N2CC(CNC(=O)Cc3cnc(C)nc3O)C2)=O)c(Cl)c1 16082,N1(C(CCS(C)(=O)=O)=O)CCC2(CC1)CC(NC(=O)C(F)(F)Cl)CO2 16083,c1(CCC)nc(C(C(=O)NCC(C)C)N(C)Cc2csc(C(F)(F)F)n2)cs1 16084,CN1CCN(C(=O)C2=NOC(CNC(=O)CN3CC(C)(C)C3)C2)CCC1=O 16085,C(=O)(C1=NOC(C)(C)C1)NC(C(=O)NCCC(C)CCO)CCF 16086,CN1CC(O)CC1C(=O)NCCNC(=O)CCCc1ccsc1 16087,CC1(C)CCC(NC(C2CC(F)(CNC(=O)COc3ccc(F)cn3)C2)=O)CC1 16088,C=C=CC(C)C(=O)NCc1c[nH]nc1C(=O)NCCCCCN(C)CC 16089,Cc1cc(CC(N2CC(C(=O)NCCNC(=O)CCCC3CC3)C2)=O)c(C)s1 16090,c1(CNC(C2C3CN(Cc4ccc(OCC)cc4)C2C3)=O)cc(C)cc(C)c1 16091,c1(C(=O)NCC(CNC(c2c(C)n(CCO)nc2)=O)C)cc(S(N)(=O)=O)cn1C 16092,c1(C(=O)NC2CCCC(N(C(CC=CC)=O)C)C2)c(F)cc(OC)cc1Cl 16093,C1(NC(CCN(CCC)C)=O)CC(O)CN(C(c2cnc(CC)s2)=O)C1 16094,C(=O)(C1CCc2c(Cl)cccc21)NC1CCN(CC2(NC(C(C=C)O)=O)CC2)CC1 16095,C(=O)(CC(=O)NC1CCC1NC(c1nnc(C(C)(C)C)s1)=O)N(C)C 16096,c1(C(N2C(C)CCC(NC(c3ccc(C(N)=O)o3)=O)C2)=O)ncn2ccccc12 16097,C1(NC(C2(CC#C)CCCC2)=O)CC2CCC(C1C)N2C(=O)CCC=C(C)C 16098,C1(C(N2CC(OC(=O)NC)C2)=O)CN(C(=O)C(C)(C)OC)CC1F 16099,C12(C(=O)NCCC3CCCC(C)C3)CC(CCO1)N(C(C1CCC1C#N)=O)C2 16100,CC(CC(N)=O)C(=O)N1CC(CNC(c2ccnn2C(C)(C)C)=O)C2(CC2)C1 16101,c1(CNC(C2(CC)CCCC2)=O)cccc(NC(=O)CC2CC(C)OC2C)c1 16102,c1(C(=O)NCC2C(NC(c3ccoc3Br)=O)C2)ncoc1C1CCCCC1 16103,Cc1cccc(F)c1CC(=O)NC1CC(NC(C2C3CCC(F)(F)C23)=O)C(O)C1 16104,N1(C(C=C2CCN(C)CC2)=O)CCC(NC(C23CCN(CC2)C3)=O)CC(C)(C)C1 16105,CC1=C(C(=O)NC2CCN(C(=O)C=C(C3CC3)C3CC3)C(C3CC3)C2)CCC1 16106,C1(F)(CNC(C2C(=O)NCC2)=O)CCN(C(c2cccc(OC(F)(F)F)c2)=O)C1 16107,C1(NC(CCC)=O)CCN(C(c2cc(N3CCCC3)nc(Cl)c2)=O)CC1C 16108,c1(CC)cccc(-n2nc(C(CC)OC)nc2-c2coc(C3CC3)n2)c1 16109,CCCCS(=O)(=O)NC(C)C(=O)NC1CC(CNC(=O)C(C)(C)NC(C)=O)C1 16110,CC1=C(C(=O)N(C)CCOCCNC(=O)CCc2cncc(Br)c2)CCC1 16111,N1(C(c2c(CC)cno2)=O)C2CCC1CC(C(=O)Nc1cnc(C)nc1C)C2 16112,CC1(NC(C2CC(NC(=O)NCc3ccccc3)C2)=O)CCC(=O)NC1=O 16113,c1(CN(C)C)cc(C(N2CC(NC(C3(C)COCCO3)=O)C(O)C2)=O)ccn1 16114,O=C(CCC(=O)c1ccccc1)NCCCN(CCO)C(c1ccns1)=O 16115,c1(CC(N2C(CNC(=O)C=CCF)CCC(C)C2)=O)csc2ccccc12 16116,C1(NC(C2CCC(C)C2)=O)CCOC2(CCN(C(C3(O)CCSC3)=O)CC2)C1 16117,O(C1CCCc2ccccc21)CC(=O)NCCCNC(C1(C)CC2CC2C1)=O 16118,C1(NC(CCCCC#C)=O)CN(C(c2cc(F)c(N)cc2F)=O)C2CCCCC12 16119,C1(C(=O)NCC(C)(C)NC(C23COCC(C2)OC3)=O)CC2(C1)C(F)(F)C21CCC1 16120,Cc1cc(NC(C)CCNC(c2nc3ccccc3s2)=O)n2nc(C)cc2n1 16121,C(=O)(C(F)(F)C(C)O)NCC(C1CCCCC1)NC(C(CCC)O)=O 16122,C1(NC(c2cc(C)c(C)[nH]2)=O)CN(C(c2ccc(O)cn2)=O)C2CCCC12 16123,CS(=O)(=O)C1CC(C(=O)NC23CC2CN(C(=O)C(C#N)C2CC2)C3)C1 16124,CCCCCC(O)CC(=O)NCC(c1ccccc1)NC(c1cc(Cl)c[nH]1)=O 16125,c1(CNC(C2C(C)CN(C(=O)C(C3CC3)C3CC3)CC2)=O)ccc2c(c1)CCC2 16126,C1(NC(C(C)c2ccsc2)=O)CCC12CN(C(c1ccc(CO)cc1)=O)C2 16127,C(Cc1cn[nH]c1)(C(=O)NOCCn1ccnn1)NC(C1CCCOC1)=O 16128,C(=O)(C(CCOC)OC)NCCC1(NC(Cc2nc(CC)sc2)=O)CC1 16129,N1(C(CCNC(=O)NC)=O)CCC(O)(C(C)CNC(=O)CNC(=O)CC(C)(C)C)C1 16130,N1(C(COCCCOC)=O)CC2CC(O)C1C2NC(C1CCCCNC1=O)=O 16131,C(=O)(C1=NNC(=O)CC1)NCCC1CC(NC(C(C(C)(C)C)N(C)C)=O)C1 16132,c1(C(=O)NCC2(C(=O)NCc3ncc(C)nc3)CC2)cccc(O)c1C 16133,CC(C)CCC(=O)C(=O)N1CCC(C(=O)NC(C2CCCC2O)C)CC1(C)C 16134,c1(C(N2CC(NC(COCCC#C)=O)C(C)(C)CC2)=O)cc(S(N)(=O)=O)c(C)s1 16135,C1(NC(c2nc(COC)[nH]n2)=O)CCN(C(C2CCC3CC3C2)=O)C(C)C1 16136,Cc1ccc(C(F)(F)C(=O)NC(C2CCCN(C(=O)CSCC(N)=O)C2)C)cc1 16137,c1(C(=O)NC(C(C)NC(C(COC)NC(C)=O)=O)(C)C)cc(N)c(Cl)c(O)n1 16138,CCC(CC)CCC(=O)NC(C1CCN(C(=O)Cn2cnc(C(F)(F)F)c2)C1)C 16139,C1(C(=O)NCC2CN(C(C=CCOC)=O)C2)(OC)CCCC(C)C1 16140,C1(C(N2CCC(N(C(C3CC(=C4CCC4)C3)=O)CC3CC3)C2)=O)COCC1C(N)=O 16141,C1(C(NOCC)=O)CCN(C(c2cnn[nH]2)=O)CC1O 16142,CCCCCCCCNC(=O)C(=O)NC(C)CNC(=O)CC1CC(SC)C1 16143,c1(C(=O)NC(c2cn(C)nc2)C(F)(F)F)nc2c(o1)CCSC2 16144,C1(C(=O)NCC=CCNC(=O)CC2CCCC2(F)F)CCn2ccnc2C1 16145,c1(C(C(=O)NCc2ccnn2C)N(C)C)ccccc1F 16146,C1(N(C(CCCO)c2cccnc2)C(C(=O)NCCC)=O)CC2CCC(C1)N2 16147,N1(C(C(C2CCC2)OC)=O)CCC(C)CC1C(=O)NC(COC)C(C)C 16148,C(C1CCc2ncnn21)N(C1CCN(C(CC(=C)C)=O)C1)C 16149,C123CCOC(C1)(C2)CNC3=O.c1(NC(C2C(=C)CC2)=O)nn(CC)cc1Br 16150,Cc1ccc(C(=O)NC(C)C(CO)NC(C2CC(S(C)(=O)=O)C2)=O)cc1C 16151,C1(C(N(C(C)(C)C)CCN)=O)CCCN1S(=O)(=O)N1CC2C(C(F)(F)F)C2C1 16152,c1(C(C)NC(C(C)N(C(=O)COC2CCCC2)CC)=O)ccc(C)cn1 16153,Cn1ccc2c(C(N3CCN(C(=O)C(C)(C)C(=O)O)C(CCCl)C3)=O)cccc12 16154,C1(CC)CN(C(C2(F)CCOC2)=O)CCN1C(=O)CCCCc1ccc(Cl)cc1 16155,n12cc(ccc1=O)CCNC(NCC(O)C)=NCC2.C(C)(C)(C)SCCSC.CO 16156,C1(NC(=O)CC2(CO)CC2)CN(C(C2CC(=O)N(C3CC3)C2)=O)CC1F 16157,C12(C(=O)NC3CC4(C(C(N(C)Cc5c(C)n[nH]c5)=O)C4)C3)CC(C)(CCO1)C2 16158,N1(C(Cn2c(C)ccc2C)=O)CCN(C(=O)COC2CC2)C(C2CCCC2)C1 16159,C=CC(CC)C(=O)NCc1cccc(CN(C)C(c2ncn(C)c2C)=O)c1 16160,C(=O)(C(C)(C)C(=O)NCC1(O)CCN(C(=O)CC2CC(C)(C)CO2)C1)NC 16161,C(c1ccc(F)c2ccccc12)=CC(=O)N(CCCNC(=O)C=C1CCSCC1)C 16162,C12(CC(=O)NCCNC(CCCCN(S(C)(=O)=O)C)=O)CCCN1CCC2 16163,C(CC(C(C)C)NC(=O)C(=O)NCC(F)(F)F)NC(CNC(C)=O)=O 16164,c1(C(=O)NC(C2CCN(C(Cc3ncc(CC)[nH]3)=O)C2)C)cc(F)cc(F)c1N 16165,CS(=O)CCC(=O)NCCN(C(=O)CN(CCO)CCO)Cc1ccc(Cl)nc1 16166,CC(C)CC(O)CC(=O)N1CCC(C)(NC(=O)CCc2ccn(C)c2)CC1 16167,C(=O)(CCS(N)(=O)=O)NCC1N(C(c2cccc(C(C)C)c2)=O)CC=C1 16168,c1(NC(C(C2CN(C(c3cc(CCC)[nH]n3)=O)C2)O)=O)ccc(C)c(C)c1 16169,c1(C(N(CCC(C)NC(c2cn(C)nn2)=O)C)=O)cccc(-c2nc(=O)o[nH]2)c1 16170,C1(CC#C)(C(N2CCC(NC(=O)CC3CCCN3C(=O)OC)C2)=O)CCCCC1 16171,CC1CC(C(=O)N2CCC2CNC(c2cncc(-c3cccc(F)c3)c2)=O)=NO1 16172,CC(C)(C)C(C(=O)NCCc1nc[nH]n1)NC(c1ccnnc1)=O 16173,c1(CC(N2C(CN(C(c3cnc(C)s3)=O)C)CCC2)=O)ccc2[nH]ccc2c1 16174,CC1CCCN1CC(=O)NCC1CCC1C(N1CCC(N2CCC2)C1)=O 16175,n1(CC(=O)NCC(CNC(CC(n2ccc(C)n2)C)=O)O)cc2ccccc2n1 16176,C#CCCC(O)C(=O)Nc1cccc(NC(=O)C(c2ccc(F)cc2)OC)c1 16177,n1(CCC)nc(C)cc1C(=O)NC(CN(C(=O)C(C)CC)C)CC 16178,N1(C(CSCC)=O)CCC2(CCN(C(c3ccc(OC)nc3)=O)C2)C1 16179,Cn1cc(C(C)(C)NC(=O)OC2CCCCC2C(N)=O)c2ccccc12 16180,c1(COC)ccc(NC(C2(C(C)NC(=O)CC3COC(=O)N3)CC2)=O)cc1 16181,c1(C(=O)NC(CC)(CNC(=O)C(C)(O)CC)CC)ccc2nc(N(C)C)oc2c1 16182,CC1(C)CN(C(c2csc(=N)[nH]2)=O)CC1C(=O)NCCC1OCCC1(C)C 16183,C1(NC(c2ccc(C)cn2)=O)CCCC12CN(C(=O)CCC1CCCCC1)C2 16184,C#CCC(C(=O)N1CCCC1(CC=C)C(N1CC(F)C(F)C1)=O)C1CC1 16185,c1(C(=O)NC(CC)CNC(C2CC(O)C2)=O)ccncc1C(F)(F)F 16186,C1(CNC(C2(F)C(C)C2)=O)CCC2(CCN(C(c3cccc(N)c3F)=O)CC2)O1 16187,CC(C)CC1C(=O)O1.c1(OCC2CCC23CCCO3)ccc(F)cc1F 16188,c1(NC(CNC(C2CC(C)(C)C2)=O)CO)ncnc2cccc([N+](=O)[O-])c12 16189,CC(C(=O)N1CCN(C(c2nccc(N)c2Cl)=O)CC1CF)C(C)(C)C 16190,C(CC(F)(F)CO)NC(=O)CC1(n2cc(-c3ccccc3F)nn2)CCOCC1 16191,C1(n2c(C(c3csc(CNC(CCCC)C)n3)C3CC3)nnn2)CCCCCC1 16192,c1(C(=O)NC(CNC(=O)CC2(O)CCOC2)C2CC2)cccn2ccnc12 16193,N1(C(=O)NCCC2CN(C(C)=O)C2)CCCCC1CC(C)C 16194,CC(O)C(=O)N1CC(C(=O)NCC2(CO)COC2)C1 16195,c1(C(N2CCCC(C(N(C)Cc3c(C)occ3)=O)C2)=O)cc2ncccc2[nH]1 16196,n1(CCCOC)nnnc1C(c1ccc(C(N)=O)o1)NC(COC)CCOC 16197,C(=O)(CC(C)C(=O)N(CC(=O)NCC1CC(C)C1)C1CC1)OC 16198,c1(-c2cc(CN(CC(C3CCCC3)OC)C)no2)ccc(Cl)cc1Cl 16199,N(C(=NCCC(C)C)N1CCc2ocnc2C1)CC(c1c(C)noc1C)C 16200,C1(C)(C(=O)NC(CCCNC(c2c(CC)n(C)nn2)=O)C)CC2(C1)CC2(F)F 16201,c1(CNC(c2c(OC)ccs2)=O)ccc(NC(=O)C(C)OCC2CCCO2)cc1 16202,c1(C(=O)NCC23OCC(NC(C4C(C=C)CC4)=O)(C2)C3)cc([N+](=O)[O-])ccc1Cl 16203,C(=O)(CC1OCCc2ccccc21)N1CCC2(N(CC(=O)NCC)CCC2)C1 16204,N1(C(CN(C)C(C2CCC(C3CC3)C2)=O)=O)CCCCCCCC1 16205,C1(C(=O)NCCCN(C(C(C)NC(COC)=O)=O)C)COCC(C)(C)O1 16206,C1(NC(C2CC3(CC3)C2)=O)CN(C(=O)CCC2CCCC2)C2(CCCC2)C1 16207,C(=O)(C#CC1CCCOC1)N1CCOCC(C)(CNC(C=CCCC)=O)C1 16208,N1(C(C2CC(=C)C2)=O)CC2C3CCC(C2C1)N(C(=O)COc1ccc(Cl)cc1)C3 16209,N1(C(C(C(CC)C)NC(C)=O)=O)CCC2(CCC2)C(NC(C2CCC(=O)N2)=O)C1 16210,C1(NC(C2(SCC)CC2)=O)COCCC1NC(c1scc(C)c1Br)=O 16211,n1(-c2ccc(C(=O)OCC)cc2)c(C)cc(CNN(CC(F)F)C(C)CO)c1C 16212,C(=O)(C1=NOC(C)(C)C1)N1C(C(C)C)(C(=O)NCCC2CCCN2C)CCC1 16213,N1(C(C(C)OCCCC)=O)CC2(NC(=O)CCn3c(C)csc3=O)CCC1C2 16214,C(=O)(C1=NNC(=O)CC1)N1CCN(C(c2c(C)nn(C)c2C)=O)C(C2CC2)C1 16215,N1(C(c2c(CC)ccs2)=O)CC2CCC2(CCNC(=O)CCC=C(C)C)C1 16216,c1(C(=O)NC2CCCN(C(=O)C=Cc3cncs3)C2)cccc2nc(O)[nH]c12 16217,c1(C(CC(=O)NCC2CN(C(C(F)OC)=O)C2)C)ccc(F)c(F)c1 16218,C1(C2CCCN(C(c3c(C4CCC4)cnn3C)=O)C2)(NC(CC(C)C)=O)CC1 16219,N1(C(c2nscc2Br)C(=O)NCCOC)CCC(=O)N(C)CC1 16220,Cc1noc(NC(C2C3CC2N(Cc2ccccc2-c2cccnc2)C3)=O)c1Br 16221,N1(C(C(CCCC)N(C)C)=O)C2CCC1CN(C(=O)C(C)=C1CC1)C2 16222,O=c1c(C(n2cc(CCNC3CC3)nn2)C)c[nH]cc1Cl 16223,CC1CCN(C(c2cc(C3CC3)ccn2)=O)C1CNC(=O)C=Cc1cc[nH]c1 16224,CCC(CC)CCC(=O)N1CCN(C(=O)CC(O)CC(C)C)CCC1C 16225,C1(N(C(c2ccc(C)cc2)C(=O)NCCC#N)CCC)CCN(C)C1(C)C 16226,C(=O)(C1CCc2nccn21)NC(C(=O)NC1(CC)CCCC1)CC1CC1 16227,C(C)(C(=O)NN1CCN(c2cccc(Cl)c2)CC1)N(S(=O)(=O)c1cn(C)nc1C)C 16228,N1(C(C(CCC)F)=O)CCN(C(=O)Cn2cc(C3CC3)cn2)CC1C1CCC1 16229,Cc1cnc(C(=O)NC2CCC(N(C)C(c3c(N)cnn3C)=O)CC2)c(C)c1 16230,C1(NC(CCc2n(C)c(S)nn2)=O)CCN(C(=O)C2=CCOC2)C12CC2 16231,N1(C(C(N)=O)=O)CCCOC(CNC(=O)CC(O)C2CC2)C1 16232,C1(NC(CCCN(CCC)CCC)=O)CCN(C(=O)CCC(=O)OC)C1CC 16233,C=CCC(C)(C)C(=O)N1CCCC(CCC)(NC(c2cc(O)nc(OC)n2)=O)C1 16234,N1(C(C(C)C2CC2)=O)CC2C(N(C)C(c3cc(-c4cccc(Cl)c4)ns3)=O)C2C1 16235,C1(CN(C(C(c2ccc(CC)s2)=O)=O)C)CCCCN1C(=O)CCSC 16236,C1(C(N2C(CC)CC(C)C2)=O)CCC2(CC2)N1C(c1c[nH]c(C)c1)=O 16237,c1(C(N2CC(CCNC(c3nc(CC)sc3)=O)C(C)C2)=O)ccc(OC)c(O)c1 16238,C12(CNC(C(=O)OC(C)(C)C)C)CCC(C(=O)O)(C1)N(CC)C2 16239,C1(C)(CNC(C=C=C(C)C)=O)CN(C(=O)CC2CCC(C)(C)O2)CCO1 16240,N1(C(C(C=C)O)=O)CC(NC(=O)CC2CCCCCC2)CC2(CCC2)C1 16241,c1(CCC)cccc(NC(=O)Cc2csc(Cl)c2)c1 16242,N1(C(C(CN(C)C)O)=O)CCC2C(CCCN2C(C2CCCCN2C)=O)C1 16243,C1(CCC(=O)NCC2CSCCO2)CCC(NC(=O)C=CCN2CCCC2)C1 16244,N1(C(C2=C(C)CC2)=O)CCC2(CC1)CC2C(N1CC2CC2C2CC12)=O 16245,C12(CNC(C3C(C)(C)C3)=O)CCC(C1)N(C(=O)CCCN1CCCC1)C2 16246,Cc1ncc(C(N2CC=C(CNC(C3CCC4C3C4(F)F)=O)CC2)=O)cc1C#N 16247,c1(NC(C)CN(C(=O)C#CC2(C)CCCO2)C)cccc(CO)c1[N+](=O)[O-] 16248,N1(CC(=O)N(C(=O)C(F)F)NC(C)C)CCN(CCc2cccs2)CC1 16249,c1(COC(C(=O)NCC(C)CN(C)C)C)ccccc1 16250,C1(NC(C#CC(C)C)=O)CN(C(C2(C#N)CCCO2)=O)CC12CCOCC2 16251,C(CC(C)C(=O)N1CC(C)(NC(=O)C(C)NC(=O)OC2CCCC2)C1)OC 16252,C=CC1(C(=O)NC(c2ccccc2F)C)CCN(C(c2ccsn2)=O)C1 16253,N(C1CCCc2occc21)C(C(CC(C)C)NC(C1CCC(=O)O1)=O)=O 16254,c1(OC)cc(CCC(=O)NC(C)CCNC(=O)CC(C)OC)ccc1F 16255,Cc1cc(C)n(C(C)C(=O)NC2CC(NC(C3CCC(F)(F)C3)=O)C2)n1 16256,c1(C(N2CCN(C(c3n(C=C)nnc3)=O)C(CCO)C2)=O)cc(F)cc(N)c1F 16257,N1(C(CCn2ccc(C)n2)=O)CCN(C(=O)CN2CC(=O)NC2=O)C(CO)C1 16258,Cc1ccc(C)c(C(N2CC(C(F)(F)F)OC(CNC(=O)C(F)(F)CO)C2)=O)c1 16259,Cc1cc(N2CCC3NC(=O)CCC3C2)nc(=NCC(F)(F)Br)[nH]1 16260,c1(C(=O)NC2C(C)CN(C(c3ccnc(S)c3)=O)CC2)cc2c(F)cccc2[nH]1 16261,c1(OC)cc(O)c(C(=O)NCC(C)N(C)C(C2CC(OC(C)C)C2)=O)cc1OC 16262,N1(C(COC2CCN(C(C=CC)=O)C2)=O)CCC(C)(C)C(OC)C1 16263,c1(OCC(=O)NCC=C(C(=O)NCCOCC)C)ccc(F)nc1 16264,C12(NC(c3cc(C)c(C)s3)=O)CCCC1N(C(=O)CCCCC(F)F)CCC2 16265,c1(CC(C)C)cccc(C(N2CC(NC(c3cn(CC4CC4)nn3)=O)C2)=O)c1 16266,C1(C)(CCC)CCN(C(C2C=CCN2C(=O)CN(C)C2CC2)=O)C1 16267,CC1CCN(C(c2cn(C)nc2C(C)(F)F)=O)CCN1C(C1CNC(=O)C1)=O 16268,CC1CC(CNC(c2cc(C3CCC3)on2)=O)CN1C(c1cn(C)c(O)n1)=O 16269,Cc1nn(C(C)(C)C)cc1C(=O)NC1CCCCC1CNC(c1cocn1)=O 16270,N1(C(C2(C)CCOCC2)=O)CCC(F)(CNC(=O)Cc2ccc(Cl)c(F)c2)CC1 16271,c1(C(=O)NC2CCN(C(C3N(C(=O)OCC)CSC3)=O)C2)c[nH]nc1[N+](=O)[O-] 16272,c1(CNC(C2CC(OC)CN2C(c2csc(CN)n2)=O)=O)c(F)cc(F)cc1F 16273,C1(NC(C(C)c2cccs2)=O)CN(Cc2ccccc2CCBr)CC1C#N 16274,c1(C(N2CC(C)C(NC(c3cccnc3C(F)F)=O)C2)=O)cnc2cc[nH]c2c1 16275,N1(C(=O)NCCc2ccc3c(c2)COC3)CCCc2cc(Br)cc(F)c21 16276,C1(C(C)O)CCN(C(=O)CNC(C)(C)C)C1C.c12ccc(cc1)Cn1cc-2nn1 16277,C#Cc1ccc(C(=O)NCC2CCN2C(c2nocc2C2CC2)=O)o1 16278,c1(C(=O)NC(CCOC)CNC(=O)COc2ccccc2Cl)cc(O)cc(=O)o1 16279,C1(C(=O)NCCN(C(=O)CC(C)(C)c2ccccc2)CCC)CC(O)C1(C)C 16280,CC1(C)CCN(C(=O)CSCC(F)F)CC1C(N1CCCC1C1CC1)=O 16281,CCCCCC(C(=O)NCC1CC1CNC(=O)CCN=c1[nH]ccs1)C(C)C 16282,N1(C(C2CN(C(C(CCC)=CCC)=O)CC(C)C2)=O)CCC(=O)N(C)CC1 16283,C(C(CC(C)C)C(=O)N1Cc2cncnc2C1)NC(C1(COC)CCCC1)=O 16284,c1(C(=O)NC)cc(=NC(=O)C2(Sc3ncccc3C)CC2)[nH][nH]1 16285,c1(C(=O)NC23CC(CNC(CCOCC#C)=O)(C2)OC3C)sc([N+](=O)[O-])cc1Cl 16286,C1(NC(c2c(C)ncnc2)=O)CC2CC1N(C(c1ccc(F)cc1Br)=O)C2 16287,c1(CNC(C(C)N(CCC)C(C2CC2(C)C(F)F)=O)=O)cccc(F)c1C 16288,C=Cc1cccc(-c2ccc(COc3ccccc3OCC)s2)c1 16289,C1(CC)CN(C(C2COC2)=O)CC1NC(c1ncccc1Br)=O 16290,c1(N2CCC(N(C(c3ccc(F)cn3)=O)CC)C2)nc(C2CCC2)nc(Cl)c1C 16291,C1(C(=O)NC2(CCNC(CCOC(C)C)=O)CCC2)CCCC1O 16292,C(=O)(C(C)CC(F)(F)F)N(C1CN(C(c2cc(C)cc(N)c2)=O)CC1(C)C)C 16293,CCS(=O)CC(=O)N1CC(CNC(C2(CO)CCC2)=O)C1 16294,N(C)(C1CS(=O)(=O)c2ccccc21)C(c1ncc(SC)[nH]1)C(=O)NCCOC 16295,N1(C(CCOCCC)=O)CCC2CCN(C(=O)CCNS(C)(=O)=O)CC12 16296,c1(NC(C2N(C(CCNC(=O)NC)=O)C(C)C2)=O)ccc(Cl)cc1C 16297,c1(C(=O)NCCC2N(C(CCCCOC)=O)CCCC2)cnc(N)c(Cl)c1 16298,C1(CNC2CCN(C(=O)NC3CCN(C)C3)CC2)CCC=CCCC1 16299,C(CCC(=O)NNC(=O)c1ccc(F)cc1Br)OC 16300,c1(C(N2CC(C(=O)OC)C(C(=O)O)C2)=O)cnc(OC)cc1OC 16301,c1(NC(C2CCN(C(C3(F)CCCCC3)=O)C2)C)ncnc2sccc12 16302,Cn1nncc1CC(=O)NC1(C(=O)NCCSCCO)CCSC1 16303,N1(C(C(CSC)O)=O)CC=CC(C(=O)N(C)CCOCCO)C1 16304,c1(OC)cccc2[nH]cc(CC(=O)NC3(O)CN(C(=O)C(C4CCC4)OC)C3)c12 16305,C1(C(=O)NC2(CF)CCN(C(c3c(C)nsc3N)=O)C2)CCc2ncncc2C1 16306,C1(NC(c2c(C)cc(Br)o2)=O)CN(C(C2CC2F)=O)CC1S(C)(=O)=O 16307,C1(CNc2nc(C(N)=O)c(Cl)cc2)CCC(c2ccccc2)=NO1 16308,C1(C2CN(C(C3CC3Cl)=O)C2)(NC(c2ccc(COC(C)C)cc2)=O)CC1 16309,c1(C(=O)NC(CNC(=O)Cc2cnccc2Cl)CO)cc(Cl)c([N+](=O)[O-])[nH]1 16310,N1(C(C(C)(C)OC(C)C)=O)CCN(C(C2CNC(=O)C2)=O)C(CCO)C1 16311,C1(C(=O)NC(CNC(C(C)OCC=C)=O)C2CC2)CCC(C)(C)O1 16312,CCCCC(O)C(C)C(=O)NCCC1CC(NC(=O)CCc2nc(CC)no2)C1 16313,N1(CCOCCS)CCNC(=O)C1.C(=O)(C(Cc1cn(CCO)nn1)NC(=O)CO)OC 16314,C1(C(=O)OC)CC12CCN(c1nnc(-c3[nH]nc(Cl)c3CO)n1C)CC2 16315,N1(C(c2c(CC)c(C)sc2)=O)CCC2(CC1)CC2NC(C1COCCO1)=O 16316,c1(C(=O)NC(C(C)NC(COCCC)=O)C)nc(C)oc1C 16317,C(=O)(C1=C(Cl)CCCC1)NCC(C(C)C)NC(C1(CN2CCCC2)CC1)=O 16318,c1(CC)cc(N)ccc1C(=O)NCC(C)CNC(=O)CC1CC(CN(C)C)C1 16319,Cc1cnc(C(N2CCC(C(C)(C)NC(c3cnc(N)c(Cl)c3)=O)C2)=O)cc1Cl 16320,C=Cn1cc(C(N2CCC(CCCCC)CC2)C(=O)NCC(=O)OC)cn1 16321,c1(CNC(C2CCN(C(CC(C)(C)C)=O)C23CC3)=O)cnc2[nH]nc(O)c2c1 16322,N1(C(c2c(OC)cncc2)=O)CC2=C(C1)CN(C(=O)C(c1cnccn1)C)C2 16323,O=C(CC(F)(F)C(F)(F)F)NC1CCC2(CC1)CN(c1ccccc1[N+](=O)[O-])C2 16324,C1(CC(=O)NCC)CC(F)CN1C(=O)Cc1csnn1.C1CC=CC1 16325,C(=O)(CCC(=O)N(C1CCCCC1NC(=O)C(=O)NCC1CC1)CC)NCCC 16326,c1(C(N2C(CCC(=O)NCC(CNC(N)=O)O)CCC2)=O)ccc2c(c1)CC2 16327,C1(NC2CN(C(C(=O)OC)=O)C(C)C2)CCCN(Cc2ccccc2)C1C 16328,C1(CNC(Cc2cnc(C)s2)=O)CC(C)CN(C(=O)CS(=O)(=O)N(C)C)C1 16329,CC1=C(C(=O)NC2CCCC(NC(c3c(N)cccc3F)=O)CC2)CCCC1 16330,C1(C(=O)NC(CNC(c2c(C)n[nH]c2)=O)(C)C2CCC2)Cc2ccccc2N1 16331,C1(C(=O)NC(CCNC(c2ccc(C(C)=O)c(F)c2)=O)C)CC2(C1)CC1(CC1)C2 16332,C1(C(N(C(C)(C)CNC(=O)COCc2nc[nH]n2)C)=O)CCc2[nH]nc(O)c2C1 16333,c1(NC(CCC2CCN(C(C(C)C3CCC3)=O)CC2)=O)cccc2cnccc12 16334,c1(C(CNC(C(CC)CC2CC2)=O)(F)F)ccc(F)cc1F 16335,C(CS(=O)(=O)N=S(C)(C)=O)NCCCCC=C 16336,C1(C)(CNC(C2C(C)C2)=O)CN(C(c2ccc(CO)c(Cl)c2)=O)C(C)(C)C1 16337,C1(C(N(C(CC)CC)C)=O)CC2(CCN(C(=O)CCC3CCCCO3)C2)C1 16338,C(C)(CNC(=O)C(C)(C)CF)(C(C)C)NC(CC(n1ccc(C)n1)C)=O 16339,C(=O)(C(F)C(C)(F)F)N1CC(C(=O)NC2CCC3(CC3)C2)(SC)C1 16340,c1(OC)ccc(C)c(C(N2CCCCC2c2cn(CCC(F)(F)Cl)nn2)=O)n1 16341,Cc1[nH]nc(Br)c1C(=O)NC(C)CC(C)NC(=O)C(C1CC1)N(C)C 16342,CC(=O)CCCCC(=O)N1CCC(NC(C2(CN(C)C)CC2)=O)CC(O)C1 16343,N1(C(C=C2C(C)(C)CCCC2)=O)CCC2CC1CN(C(=O)C(O)c1ccsc1)C2 16344,S(=O)(=O)(c1cccc(C(N2CC(=O)NCC2C)=O)c1)NCC(C)O 16345,c1(C(N2C(CNC(C3CC4CC4C3)=O)CC(C)(C)C2)=O)cc2ccnc(Cl)c2[nH]1 16346,c1(N)ccc(C2=CCN(N(C)C)CC2)cc1.C1(C)CC1 16347,c1(OCCOCC)ccccc1C=CC(=O)OC(C)Cc1ccccn1 16348,C1(CNC(C(C)(C)C)=O)Cc2ccccc2CN1C(C1CC(S(C)(=O)=O)C1)=O 16349,C1(C(=O)NCC(CNC(COC(CC)(C)C)=O)(C)OC)OC(C)(C)OC1(C)C 16350,N1(CC(=O)NCC(CC)N(C)C)CCN(C(=O)C(C)CCN(C)C)CC1 16351,Cc1cc2ccc(C(=O)NCC3CN(C(c4cocc4C)=O)C3)cn2c1 16352,C=C=C(C)CC(=O)NC1(CN(C)C(C2CCN2C2CCCC2)=O)CC1 16353,N1(C(CN2C(C)CC2)=O)CC2=C(C1)CN(C(=O)CN(c1c[nH]nc1Br)C)C2 16354,C(=O)(C(F)(F)C(O)C(C)C)N1CC2(C(NC(c3cccc(C)c3F)=O)CCC2)C1 16355,C1(C(=O)NC2(CCNC(C3(C(=O)NC)CC3)=O)CC2)CC(=O)CC12CCC2 16356,c1(C(N2CCN(C(C)C(=O)NCC(F)(F)F)CC2)=O)nccn2nccc12 16357,c1(C(=O)NC(C)Cn2ccnc2)cccc(CNC(C2OC3CCC2C3)=O)n1 16358,Cc1c(Cl)ccc(C(N2CCOC(C)(CNC(=O)C(C)OCC(C)C)C2)=O)c1O 16359,c1(C(=O)NCC2(C)CCCN2C(=O)C#CC2CCCO2)cccc2c1OCCC2 16360,N1(c2c(C#N)cncc2)CCC2C(CCCN2C(=O)CC2(O)CCOC2)C1 16361,C1(OC)CCCCC1(c1nnnn1CCC1CC1)Nc1cn[nH]c1 16362,C1(C(=O)Nc2ccns2)CC2(CCN(Cc3cc(O)cc(Cl)c3)CC2)C1 16363,C1(O)(CCNC(Cc2ccc(OC)cc2)=O)CCN(C(=O)Cc2cnns2)CC1 16364,c1(OC)ccnc(N2C3CN(C(=O)C(CO)NC(=O)OC(C)(C)C)CC23)n1 16365,N1(CC(=O)NCC2N(C(Cc3nc(C)[nH]n3)=O)CC=C2)CCCCS1(=O)=O 16366,N1(C(COCCC)=O)CC2COCCC2(NC(c2cc3sccc3[nH]2)=O)C1 16367,C(=O)(NN1CCCC(C(=O)CCN2CC3CC3C2)C1)c1cnc(C)[nH]1 16368,n1(CC)cc(Cl)c(C(N2CC(CNC(=O)CC(C)(F)F)CC2C)=O)n1 16369,C1(C(N2C3(CNC(C4CC(OC)C4)=O)CC(C2)C3)=O)CC12CCC(=O)CC2 16370,C1(C(C)C(=O)NCC(F)Br)CCN(C(C2CC(=O)C2)=O)C1 16371,C(CCCCN(C)C(C1(Br)CC1(C)C)=O)NC(C(C)C1(O)CCC1)=O 16372,N1(C(=O)C2=CCCC2)CC2(CO)CC1(C(=O)NCC1CC(O)CCO1)C2 16373,N1(C(c2cnn(CC)c2C)=O)CCC(NC(=O)CCn2ccccc2=O)C(C)C1 16374,N1(C(c2cc(C(F)F)[nH]n2)=O)CC2(CCN(C(C3CC(CC(F)(F)F)C3)=O)C2)C1 16375,C1(C(=O)NC(CC(=O)OCC)C)CCN(C(c2c(C)cnn2C)=O)CC1(C)C 16376,Cc1cc(Cl)ncc1CC(=O)NC1CCC(NC(c2nc(Cl)c(Cl)s2)=O)C1 16377,C=C(C)CC(C)C(=O)N1CC2CC2(CNC(=O)CCC=Cc2ccccc2)C1 16378,c1(C(N2C(CN(C(c3nc(Cl)oc3C)=O)CC)CCC2)=O)cnn2ccsc12 16379,N1(C(CCC2N(C)CCCC2)=O)CCN(C(=O)CCCF)C(CC2CC2)C1 16380,c1(OC)ccc2cc(C(=O)NC3CC3NC(=O)C(C)(C)CC(C)(C)C)n(C)c2c1 16381,N1(C(CN2C(C)CCC2)=O)CCC(C(=O)Nc2cccnc2Cl)CC1 16382,Clc1ccc2ccc(=NCCC34CCC(CC3)CO4)[nH]c2c1 16383,C1(NC(C2CC3CCCC23)=O)CCCNC12CC2 16384,c1(C(=O)NC2CCN(C(c3cc(Cl)sc3Cl)=O)CC2)cc(Cl)nc2ccccc12 16385,c1(NC2(COC)CCSC2)ccc(S(=O)(=O)NCC(CO)C(C)C)cc1Cl 16386,c1(-c2cn(CC(C)NC(C3C(CC)OCC3)=O)nn2)ccc(Cl)cc1Cl 16387,c1(C(=O)NCCOCCNC(C2(C)CNC(=O)C2)=O)cc(Cl)cc(F)c1F 16388,N1(C(CC)=O)CCC(C)C(CCNc2cc(C(=O)OC(C)(C)C)cc(CC)c2)C1 16389,c1(CCC)ncc(C(=O)NC2CC(CNC(c3cn(CCO)nn3)=O)C2)s1 16390,C1(CNC(=O)OC(C)(C)C)CN(C(=O)Cc2cn[nH]c2)CC1O 16391,C1(NC(C2(SC)CC(O)C2)=O)CN(C(=O)CSc2cccc(Cl)c2)CC1(C)C 16392,C(N=c1[nH]cnc2c(Br)nn(C)c12)C1CN(C(C=NOC)=O)C(C)C1 16393,c1(C(C)C)cc(C(=O)NCC2CCC2NC(C2(C#N)CCC=CC2)=O)cc(F)c1 16394,N1(C(c2cc(OCC)n[nH]2)=O)CC(C(=O)NC2CC(CN(C)C)C2)C(C)C1 16395,CCCCCCCCC(F)C(=O)NC(C)CNC(c1cnc2ccnn2c1N)=O 16396,c1(CC)ccc(C(=O)NCC2CC(F)(F)CN2C(c2cc(C)sc2C)=O)c(F)c1 16397,C12(CNC(C=CSC)=O)CCC(CC1)N(C(c1cc[nH]c1)=O)C2 16398,c1(C(=O)NC2(COC)CCN(C(C(CCC)OC)=O)C2)cncc2ccsc12 16399,c1(C(=O)NCC(CC=C)NC(=O)CCc2cncs2)n[nH]c2c1CC(C)OC2C 16400,c1(C(N(CC(CNC(C(c2cccc(C)c2)F)=O)C)C)=O)cccc(C)c1O 16401,C(=O)(CC(C)CNC(c1ccccc1CC#N)=O)NCC(=C)Cl 16402,c1(CCCC(=O)NCCCNC(CSCCC(C)C)=O)cc2ccccc2o1 16403,c1(NC(c2nc(NC(C3N(C(C)=O)CC(O)C3)=O)sc2)=O)c(C)ccnc1C#N 16404,c1(C(N2CC(CNC(C(CC)CO)=O)C(C)CC2)=O)cn2cnnc2cn1 16405,C1(NC(=O)CN2CC(C(F)(F)F)CCC2=O)CCCCN(C(C2CCC2)=O)CC1 16406,C1(NC(C=COC(=O)OC)=O)C2CCC(C2)N1C(c1cc(OCC)ccc1Cl)=O 16407,N1(C(CSC)=O)CC(CCNC(C23CCC(CC2)OC3)=O)OC(C)C1 16408,c1(N2C(C)CCN(C(c3cccc(F)c3Cl)=O)CC2)nc2c(cc1Cl)C(=O)OC2 16409,c1(OC)ccnc(OC)c1C(=O)NCC1(NC(C2COC(=O)N2C)=O)CCOC1 16410,Cc1ccc(F)cc1N(C)C(C1C2CN(C(c3cncnc3)=O)CC12)=O 16411,C1(N(C(=O)CC2CCCCC2)C)CC2CC1N(C(c1c[nH]cc1C(F)(F)F)=O)C2 16412,C1(CC#C)(C(=O)N(C(C)CNC(=O)Cc2ccnn2C(C)C)C)CCCCO1 16413,N1(C(C2CC(CC)C2)=O)CC(C(=O)NC23CCCC2OCC3)C(C)(C)C1 16414,c1(C(=O)NC2CCN(C(C3CC(C(F)F)C3)=O)C2)ccc(CO)c(Cl)c1 16415,C(N=c1[nH]c(=NCCC(F)(F)Cl)[nH]c2ccc(Cl)cc12)c1scc(COC)c1 16416,c1(SC)ncc(C(=O)NCCC2(O)CN(C(c3csc(F)c3)=O)C2)n1C 16417,c1(C(N2CCC(NC(CC(CCC)O)=O)CC(O)C2)=O)cnc2c(cnn2C)c1 16418,C#CCCCCC(=O)N1CCN(C(C2(C)CCOC2)=O)CC1C(F)F 16419,N1(C(c2n(CCC)nc(C)c2)=O)CCCCC(CNC(=O)CC2CC(SC)C2)C1 16420,N1(C(c2cc(N3CCOCC3)ncn2)=O)CCC(C2CC2(F)F)C1 16421,CCC(F)(F)C(=O)NCc1ccccc1N1CCN(C(C2(C#N)CC2C)=O)CC1 16422,c1(C(=O)NCC(O)CCNC(C2CCCCCCC2)=O)cncc2c1CCCC2 16423,C1(N(C(C=C(C)C(F)F)=O)C)CCC2CN(C(=O)Cc3ccsc3C)CC12 16424,N1(C(C2CC(F)CN2C(=O)Cc2cccc(F)c2F)=O)CCCC2(CCO2)C1 16425,C1(CNC(C(CCOC)(C)C)=O)CC2COCC2N1C(=O)Cn1ncn(C)c1=O 16426,N#Cc1ncn(CC(=O)NCC2CCC(NC(=O)Cc3ccn(C(F)F)n3)C2)n1 16427,C(CNC(c1nscc1C)=O)(CC(=O)NCCN1CC2CCC1C2)OC 16428,c1(-c2ccccn2)ncc(OCCn2cc(C3CCCO3)nn2)cn1 16429,N1(C(CC2(NC(C)=O)CC2)=O)CCCN(C(C2CCS(=O)(=O)N2)=O)C(CO)C1 16430,C=CCCCN(C)N1CCCC(N(C)C)C1 16431,c1(C(N2C(C)CCC(NC(c3c(CC)cns3)=O)C2)=O)ccc2cnncc2c1 16432,c1(C(=O)NCC2(CCNC(CSc3n(C)ccn3)=O)CC2)cc(S(C)(=O)=O)cs1 16433,N1(C(Cc2cn(CC)nn2)=O)CCC2(CCC2)C(CNC(c2cn[nH]c2)=O)C1 16434,C(=O)(C#CC(C)(C)CNC(c1c[nH]c(C)c1)=O)NC1CCCN(CC)C1 16435,C(=O)(C(C)CC(C)C(C)=O)N1C(C)(CC(=O)NCC=CCSC)CC1 16436,Cc1cc(C(=O)NCC2CCC(CNC(C34CCCCC3C4)=O)CC2)ccc1F 16437,C1(C(N2CCC(N(C(=O)CCSCC)CCC)C2)=O)CC(F)CN1C 16438,C(=O)(CCCC(OC)OC)NCc1c(NC(CC(CC)OC)=O)cccc1 16439,C1(CNC(c2c(C)onc2Cl)=O)CN(C(C2CCC(=O)C2)=O)CCC1(F)F 16440,C1(CCC(=O)NC(C)(CNC(c2ccc[nH]2)=O)C2CC2)CCCCO1 16441,c1(C(=O)NC(C)CCCCNC(=O)C(C)(O)C2CCC2)cn(C)c(=O)nc1O 16442,Cc1cc(F)c(C(N2CCN(C(=O)CCS(C)(=O)=O)CCC2C)=O)cc1F 16443,N1(C(CC2CC(C)(C)OC2)=O)CCC2CN(C(c3ccncc3)=O)CC2C1 16444,n1(CCCC)nccc1C(N1CCC(C(C)NC(c2cncnc2)=O)C1)=O 16445,N1(CC(C)NCCCC)Cc2ccccc2C(C(=O)OC(=O)CC)C1 16446,Cc1cc(CC(=O)NC2(CF)CCN(C(C3CCS(=O)(=O)CC3)=O)C2)cc(F)c1 16447,c1(SCCC)ccc(C(=O)NC(C)CCCNC(c2cn(C)nc2CC)=O)cc1 16448,Cc1cc(C)c(C(=O)NC2CC(NC(=O)C(O)CC(F)(F)F)C2)c(O)n1 16449,C(C(c1nnnn1CC1CCOCC1)Nc1cccc(CCO)c1)(C(C)C)OC 16450,CC(C(CO)NC(=O)CC(C)NC(=O)OCc1ccccc1)NC(C1CC1F)=O 16451,C1(C)(CNC(CCc2c(C)ncs2)=O)COCCN(C(=O)C(C)C(F)F)C1 16452,N1(C(CC2(C)CC2)=O)CC2CCC2(NC(=O)CCc2ccc[nH]2)C1 16453,CC1(O)CCC(CC(N2CC(F)(F)CC2CNC(C2CCS(=O)(=O)N2)=O)=O)CC1 16454,c1(C(N)=O)nc(NC2CS(=O)(=O)CC2CC2CC2)cc(C2CC2)n1 16455,Cc1ncc(C(N2CC3(CCN3C(=O)Cc3ccoc3)C2)=O)c(Br)c1Cl 16456,C(=O)(C#CC1(C)CCCO1)N(C)CC1CCCN1C(c1cc(F)cnc1Cl)=O 16457,C12(C(N3CCC(COCC)C3)=O)CC(CO)(CN1C(=O)CCNC(C)=O)C2 16458,c1(C(N2CC(CN(C(=O)C(N)=O)C)OCC2)=O)cn2ccsc2n1 16459,C1(NC(CN(C(=O)CN2C(C)CCC2C)CCOC)=O)C(C)CCC1C 16460,Cc1ccc2nc(C(=O)NCCCCNC(c3ccc(C)cc3C)=O)c(N)n2c1 16461,C1(OC)CCCC(C(=O)NCC23CC2CN(C(=O)C(CCSC)OC)C3)C1 16462,CC1CN(C(c2cc(F)c[nH]2)=O)CC(C)N(C(c2cc(Cl)c(F)cc2O)=O)C1 16463,c1(CC(=O)NCC2C(NC(C(C)OC)=O)CC2)cc(C)nn1C 16464,C#CCC(O)C(=O)NCC1C=CC(NC(C2(C(c3ccccc3)=O)CC2)=O)C1 16465,N1(C(c2c(OCC)cccn2)=O)CC2CC(NC(=O)C(=O)N(C)C)C2C1 16466,C(=O)(NNc1cc(F)ccc1C(F)(F)F)c1c(Cl)ccc(NC(CC(C)C)=O)c1 16467,C1(NC(C(CC)O)=O)CN(C(c2cc(C(C)C)ccn2)=O)CC1(F)F 16468,c1(OCC=C)ccc(S(N)(=O)=O)cc1C(N1CCC1CNC(=O)C(O)C1CC1)=O 16469,c1(C(COC)N(CC(C)C(=O)OC(C)(C)C)C(=O)C(C)(C)C)cccc(Cl)c1.C1(=O)CC1=O 16470,C=C1CON(C(=O)COC2CCN(C(=O)C(O)C(C(C)C)OC)C2)C1 16471,c1(C2(C(=O)OC)CC2)ccc(-c2ccc(SCCN3CCN(C)CC3)cn2)cc1 16472,Cc1ccc(C(c2nnnn2C)NCC2(C(F)F)CCCO2)cc1 16473,C1(NC(C(C)(O)C2CCC2)=O)CC2CCC(C1)N2C(=O)CCc1nc(=N)[nH][nH]1 16474,c1(C(=O)NC2C3CN(C(c4n(CC)ccc4)=O)C2CC3)nc(C)c(N)cc1C 16475,C(CC(C(=O)N1CCC(C)(CN(C)C)C1)NC(=O)COC)=CC 16476,C1(NC(c2ccc(CSC)cc2)=O)CC2CN(C(C3(C)CCCC3)=O)CC12 16477,C1(CNC(COC(CC)CC)=O)CCCN(C(c2nnsc2C)=O)CC1 16478,N1(C(C)C)CCC(C(=O)NCC2CCCN2C(C2CCCC3CC23)=O)CC1 16479,Cc1ccc(I)cc1CN1CCS(=O)CC1c1cnn(C)c1 16480,N1(C(=O)C2=CCCO2)CCCC2(C1)CN(C(C1C3C4CCC(C4)C13)=O)CCO2 16481,c1(C(N(C(C)C(=O)NCc2cc(O)cc(F)c2)CCC)=O)cnn2cccc2c1 16482,Cn1c(C(=O)NCCCCC(CO)NC(c2cnc[nH]2)=O)c2n(c1=O)CCCC2 16483,CCCC(C)CC(C)(c1nnnn1C(C)C)Nc1ccc(C(=O)N(C)C)c(C)c1 16484,C12(NC(CCCCC(N)=O)=O)CN(C(=O)CCN3CCCC3)CC1CS(=O)(=O)C2 16485,CC(CC(=O)NC1CCCN(C(c2ccc(C3CC3)cn2)=O)CC1)C(F)F 16486,CC1CCN(C(=O)CCc2nncs2)CC1NC(C1CCN(C(=O)N(C)C)CC1)=O 16487,CCCC(CC)CC(=O)N1CC(CO)(NC(=O)CNC(=O)Nc2ccccc2)C1 16488,N1(C(c2[nH]nc(OC)c2Cl)=O)CCC2(NC(=O)Cc3cscn3)CCCCCC12 16489,c1(C(N2C(C(N)=O)COCC2)=O)cc2c(OC(F)F)cccc2[nH]1 16490,C(=O)(C(C)P(C)(C)=O)NC1CCC(NC(c2cncc(NC(CC)=O)c2)=O)CC1 16491,Cc1cccc(C(CN2CCCC(C)C2)NCCCC(C)(C)N(C)C)c1 16492,CCCC(COC(=O)C(CC)OC)CCO 16493,S(=O)(=O)(c1ccc(NCC2CCCC3(CCOC3)O2)c(Cl)c1)NCCCCCC 16494,c1(OC)ccc(C(N2CCCC(C)(CNC(C3(SC)CCC3)=O)C2)=O)cc1Cl 16495,CC1CC(C(N2CCCC2CNC(c2occc2C2CC2)=O)=O)CC(C)C1 16496,c1(CNC(C2CC2Cl)=O)cccc2c1CN(C(c1ccn3nnnc3c1)=O)C2 16497,c1(C(=O)NCC2CCC(NC(CN3CCC(C)C3)=O)C2)ccc2nc(O)[nH]c2c1 16498,N1(C(Cc2scc(C)c2)=O)CCCC(C(C)NC(=O)C(C)(C)n2cccn2)C1 16499,Cc1nc(C)c(F)c(=NCCOc2ccccc2NC(=O)C(C)(O)C(C)C)[nH]1 16500,CC(CC(C)(C)C)NC(=O)C(c1cccs1)NC(=O)CC1NC(=O)NC1=O 16501,C(=O)(CCCCC(C)CC)N1CCC(C)(CCNC(c2c(CC)noc2C)=O)C1 16502,c1(CC(=O)NC2CC(NC(C3(COC)CC3(C)C)=O)C2)ccnc(C(=O)OC)c1 16503,N1(C(c2n(CC)cnn2)=O)CCN(C(c2coc(C(C)C)n2)=O)C2CCCCC12 16504,C=C1CCN(C(=O)CSCCCOC)C(C(=O)NC(C)Cn2ccnn2)C1 16505,C1(CC(=O)NCC2COCCN2C(=O)CC2CCCCC2)CCC(F)(F)CC1 16506,N1(C(C(C(C)C)C)=O)CC(CNC(c2cc3ccccc3o2)=O)OC(C)(C)C1 16507,N1(C(c2n(C)ncc2Br)=O)CC2CCC2(CC(=O)O)C1.C1(N)CCC1 16508,C1(C(=O)NC(CCCN(C(=O)OCCC(=O)OC)CC)C)Cc2ccncc2C1 16509,c1(CC(C=C)O)cn(CCCC(=O)N2CC(CS(C)=O)C2)nn1 16510,C1(CNC(c2c(C)scn2)=O)CC2CCC1N2C(C1(C)CC(F)C1)=O 16511,CC(CC1CC1)C(=O)NCC(C)(C)NC(=O)C(C)n1ccnn1 16512,C1(C(=O)N2CCC(c3ncco3)C2)(C(CC)=O)CCCc2ccccc21 16513,CS(C)(=O)=NC(=O)C(=O)NC1CC(c2ccccc2)(NC(=O)COC(F)(F)F)C1 16514,C1(CNC(C(COC)N(C)C)=O)CN(C(=O)CC2CN(C(C)=O)C2)CCN1C 16515,O=C1NCC2(CCN(C(C3CCOCC3NC(=O)C(O)CC3CCCC3)=O)C2)N1 16516,C(=O)(CC(C)NC(=O)CC1(C)OCCO1)NC(CC#C)C 16517,N1(C(CS(C(C)C)(=O)=O)=O)Cc2nccn2CC(NC(=O)C=C2CCC(C)C2)C1 16518,C(c1cccc(CO)c1)=CC(=O)NCC(C)NC(c1ccnc(C(F)F)c1)=O 16519,c1(OC)ccc(C(=O)NC2CCCCC2NC(c2ncc(N)nc2C)=O)c(Cl)c1 16520,Cc1cc(C(=O)NC(C)(C)CC=CC(=O)NC(C)C(C)CO)n[nH]1 16521,CCC(CC(=O)N1CCC1CNC(c1ccc(CSCC)s1)=O)c1ccccc1 16522,N1(C(c2c(C)noc2C)=O)CC2(C1)SCCC2NC(=O)C(O)C1CCCC1 16523,CC(Cc1cccs1)N=c1ccnc(N2CCOCC(C)(F)C2)[nH]1 16524,c1(OC)cc(Br)cnc1C(=O)NCC(C)CNC(c1cnn2c1OCC2)=O 16525,c1(C(=O)NC(C(C)NC(=O)C=Cc2cc[nH]c2)C)cc2cc(Cl)cc(Cl)c2[nH]1 16526,c1(CC(=O)NCCNC(c2ccn(CC)c2C)=O)ccc(C)cc1C 16527,C1(NC(CCCNC(=O)Cc2cccnc2O)=O)CCOC12CCOC2 16528,N1(C(C2(CC#C)CCC2)=O)CC(NC(c2ccc(C(F)(F)F)s2)=O)CC2(CC2)C1 16529,CC(=O)CCCC(=O)NC(C)(CNC(c1nccc(Cl)c1Cl)=O)C1CC1 16530,n1(CCNC(C(C)C2(O)CCC2)=O)ccc(C(=O)NC2(C(F)(F)F)CC2)c1 16531,CC1CN(C(=O)C=CCF)CC1NC(C1(c2cccc(Cl)c2)CCCCC1)=O 16532,CCCC(=O)NNC(=O)C(=O)Nc1cccc(N=[N+]=[N-])c1 16533,C(=O)(CCCCCCn1cc(-c2cscn2)nn1)N(C)CCc1cccnc1 16534,C(C)(C)(CCN=c1[nH]cnc(C)c1Br)NC(COc1c(C)occc1=O)=O 16535,CC(C)(C(=O)N1CC=CC(C(=O)NCC(CO)C(C)(C)C)C1)C(F)(F)F 16536,C#CC1CN(C(c2cc([N+](=O)[O-])n[nH]2)=O)CCN1C(=O)C=C(C)c1cccs1 16537,C1(CNC(CC2CC(CC)C2)=O)CN(C(=O)CSC2CC2)CC1C(F)(F)F 16538,CC(CCC(F)(F)F)NC(=O)CC(C)(C)NC(=O)Cc1ccsn1 16539,C(=O)(C1=CCCCCC1)NCc1ocnc1CNC(=O)CC1NC(=O)NC1=O 16540,c1(C(C)C(=O)NCC2(O)CN(C(=O)CSCc3cc(Cl)no3)C2)ccc(F)cc1 16541,Cn1cc(CN2CCC(NC(c3cncc(-n4cccn4)n3)=O)C2)c(Cl)n1 16542,CCC(CC(F)F)C(=O)N1CCC(CN(C(=O)C(C)c2ccco2)C)C1 16543,c1(SC)nc(C)c(CC(=O)NCC23CCCC2CCN3C(=O)C(N)=O)c(O)n1 16544,C1CC(=O)NNc2ccccc2-c2nc1n(CC)ccccc2 16545,C1(NC(CS(C)(=O)=O)=O)CC(NC(=O)CCCn2cnc(C#N)n2)C12CCC2 16546,C(=O)(CC1=CCCCC1)N1C(CNC(c2ccc(C(C)=O)c(O)c2)=O)C(C)CC1 16547,c1(C(N2C3C(NC(C=CC)=O)C(CC3)C2)=O)sc2ccccc2c1CS(C)=O 16548,Nc1nc(C(N2CCC3(NC(=O)COC(F)F)CC3C2)=O)ccc1O 16549,C1(c2nc(C)[nH]n2)CCC(CNC(N2CCOCC2c2ncnn2C)=O)CC1 16550,c1(C(N2CCC(N(C(C=CC=CCC)=O)CC)C2)=O)csc(=NC2CC2)[nH]1 16551,N1(C(c2cn(CC)nn2)=O)CCC(NC(=O)CCc2cccc(C)c2)C(CO)C1 16552,C(C1=CCN(C(=O)OC(C)(C)C)C1)Sc1occ(NC(C)=O)n1 16553,CCC(C)(C)C(=O)N1CCC(N(CCO)C(C2CCC(C)(C)O2)=O)C1 16554,c1(C2(CNC(N(C3CC(C)=NO3)CCC)=O)CC2)cc(Cl)ccc1C 16555,C12(C3CCCN(C3)C(=O)N1)CC2.C1(C)(CC(=O)OC)CC(OC(C)(C)C)C1(F)F 16556,CN1CCCC2(CCN(C(CC3CCC4CC34)C(=O)NC(C)(C)C)C2)C1 16557,N1(C(c2ncccc2C(F)(F)F)=O)CCN(C(c2cn[nH]c2)=O)C(CC2CC2)C1 16558,N1(C(C2CC3(CCCCC3)C2)=O)CCn2ncc(C(N3CCC(Cl)C3)=O)c2C1 16559,N1(C(c2onc(CC)n2)=O)CCC(C)C(CNC(=O)CCCCF)C1 16560,c1(C(=O)NC2CN(C(C3CCCC3O)=O)C2)cccc(O)c1Cl 16561,N1(C(CCSCCC)=O)CCOC(CN(C(=O)CN2CC(C)(OC)C2)C)C1 16562,Cc1ccc(C(N2CCC(F)(C(=O)NCCCC(O)CO)CC2)=O)nc1C 16563,C1(CCC)CN(C(C2OCCC2C)=O)CC1C(=O)N(C)Cc1ccn(CC)n1 16564,CCC(C)(CNC(=O)COC1CC(NC(=O)CCC2CCCCO2)C1)CC 16565,C1(O)(C(=O)NCC2CC(NC(Cc3ccn(CC)n3)=O)C2)CCCC(C)(C)CC1 16566,Cc1ocnc1CC(N1CSCC1C(=O)NOC(c1ccncc1)C)=O 16567,N1(C(C)=O)CCCC1CC(N1CC(O)(CCNC(=O)C(C)(C)c2ccno2)C1)=O 16568,C(=O)(C1=NOC(C)C1C)NCC1(NC(c2cc(F)cc(Cl)c2N)=O)CC(OC)C1 16569,CN1CC(N=c2nc3c(cnn3C)c(NCCc3c[nH]c4ccc(F)cc34)[nH]2)C1 16570,c1(N(C)Cc2ccc(C)cc2)nc2c(c(=NCC(C(C)C)C(C)C)[nH]1)SCC2 16571,C(=O)(C1=Cc2cc(Cl)ccc2OC1)NC1C2CN(C(Cc3cc(C)[nH]n3)=O)C1C2 16572,CC(C)(CC(F)C(=O)NCCC1CCCC12CC2)NC(C1CC2CC2C1)=O 16573,c1(C(N2CC(NC(C3(C(F)F)CC3)=O)CC(O)C2)=O)ccc2ncccc2n1 16574,c1(C(=O)NC(C2(NC(=O)CC3CCCC(O)C3)CCCCC2)C)cn2c(n1)CCC2 16575,C(=O)(CCCN=[N+]=[N-])NCCOCCCNC(C1(OC)CCCC1)=O 16576,C1(CNC(c2coc3c2COC3)=O)CN(C(=O)C=CBr)C2CCN1C2 16577,c1(C(N2CC(c3n(C)cnn3)OCC2)=O)ccc(OC(F)F)c(F)c1 16578,c1(C(C(=O)NC(=O)OC(C)(C)C)N(C2COCC2CC)CC2CCC2)ccnc(O)c1 16579,C1(C(=O)NCC2(F)CC(NC(C3(CC(C)C)CC3)=O)C2)CCC2C(C1)C2(F)F 16580,C1(NC(c2cc(C)c(-c3ccc(F)cc3)s2)=O)CN(C(=O)CC(F)F)CC1(C)C 16581,C1(NC(C2(C(=O)OC)CC2)=O)CC2CCC1CC2NC(c1cc(Cl)ncc1OC)=O 16582,N1(C(C(CC)=O)=O)CCC2CC(C(N3CCC(F)(CO)CC3)=O)C2C1 16583,C(C)(C)(C(C)CC(=O)NC1CCCC1(C)O)OC 16584,N1(C(C=CC(C)(C)C)=O)CC2(C1)SCCC2NC(=O)COC1COC1 16585,C1(N(C(C=CC(CC)=CC)=O)C)CN(C(=O)Cn2ncc(Cl)c2C)CC1(C)C 16586,Cc1nnccc1C(N1CC(C(C(=O)Nc2ccc(SCCCO)cc2)O)C1)=O 16587,N1(C(C2C(=C)C2)=O)CCC2CN(C(=O)CCCc3nncn3C)CC12 16588,C1(C(=O)NCC2(C)OCCO2)(NC(c2ccccc2)=O)CCCCC1 16589,Cc1nn(CC(=O)NC2CC(C)N(C(C34CCC(C3)C4)=O)C2)cc1Cl 16590,CC1(C)C(C(=O)NCC2CN(C(=O)C(C)(C)c3sccc3Cl)CCO2)C1(C)C 16591,NC(CC(=O)N1CCCCC1Cc1ccccc1F)C(=O)O 16592,c1(OCC)c(Br)cc(N(CC)CC)cc1S(=O)(=O)N1CCC(C(C)CO)CC1 16593,Cc1cnc2n1CCC(NC1CCS(=O)(=O)CC1)C2 16594,c1(OC)ccc(C(=O)N(CC(C)(C)CNC(=O)Cc2cc[nH]n2)C)c(F)n1 16595,S(=O)(=O)(c1cc(C(=O)NC(C)CNC(=O)C(C#N)C(C)C)ccc1F)NCC=C 16596,N1(c2snc(C)c2C#N)CC2CCC1C1CN(C(=O)CSc3ncccn3)CC21 16597,C(C(C)(O)CC(=O)NC1CC(NC(c2nc(C)n(C)c2C)=O)C1)OC 16598,c1(CC)[nH]nc(C(=O)NC(CNC(c2ccnc(S)c2)=O)C(C)(C)C)c1C 16599,c1(C(N2CC=C(CNC(c3c(F)ccc(C)c3)=O)CC2)=O)cccc2c1NCC2 16600,O=C1CN(C(=O)CCC2CCN(C(=O)Cc3ncccc3F)CC2)C2(CC2)CN1 16601,C(=O)(CCC(C)NC(C1CC(O)C(F)C1)=O)NC1(C(=O)OC)CC(C)C1 16602,c1(C(=O)NCC2CC(C)N(C(=O)CN=S(C)(C)=O)C2)cc2c(F)ccc(F)c2[nH]1 16603,c1(C(=O)NCC(C(C)(C)C)NC(c2cnc(S)[nH]2)=O)cc(O)ccc1Br 16604,C1(C(N(C2(C(N3C(C(=O)OCC)CC(O)C3)=O)CC2)C)=O)CCCCN1N=O 16605,N1(C(=O)Cc2cocn2)CC2CN(C(C3CC4C=CC3C43CC3)=O)CC2C1 16606,C(=O)(C(CC(C)C)C(C)C)NS(CCCOC1CN(S(C)(=O)=O)C1)(=O)=O 16607,N1(C(C2CC(=C)C2)=O)CC(N(C)C(c2cccc(F)c2C)=O)C(C)(C)C1 16608,C(=O)(C1=NOC(C)C1)NC(C(=O)NCC(C(F)(F)F)OC)C1CCC1 16609,NS(=O)(=O)c1cccc(C(=O)OCc2nc(CO)cs2)c1 16610,C(=O)(C1=CCC2CCC1N2C(=O)C(C#N)C(C)(C)C)NCC=CC=CC 16611,C1(OCC)CC2(C1)CC2C(=O)NCCN(C(=O)CC1CC2C=CC1C2)C(C)C 16612,C1(C(=O)NC2(C(=O)NCc3ncc(C)cn3)CCN(C)C2)CC2(CCC2O)C1 16613,N1(C(COC(CC)(C)C)=O)CC(C(N2CCOC(C3(C)CC3)C2)=O)C(F)C1 16614,CN=c1[nH]c(C(N2CC(C(C)NC(C3CCN(CC(F)(F)F)CC3)=O)C2)=O)cs1 16615,c1(OC)ccc(C(C(=O)O)NC(C2CCCCC2(F)F)=O)cc1Cl 16616,C(=O)(C(CNC(c1cc(C(N)=O)[nH]n1)=O)OC)NCC(=C)Cl 16617,C1(O)(C(CNC(C(C)N(C)C)=O)C)CCN(C(=O)Cc2sccc2Cl)C1 16618,N1(C(C(c2ccccc2)OCC(C)C)=O)CC2(CCCN(C(=O)C(C)SC)C2)C1 16619,Cc1ncccc1C(=O)NC1CC(O)(CNC(C2CC3(CSC3)C2)=O)C1 16620,C(=O)(C(C)CCCOC)N1CCC(OCCCNC(C(C)OCCC=C)=O)CC1 16621,c1(C(=O)NC2(CC=C)CCN(C(=O)C(C)S(N)(=O)=O)C2)c(OC)cccc1OC 16622,c1(C(N2CC(NC(C3CN(OC)C(=O)C3)=O)C(C)C2)=O)nccn2cc(C)nc12 16623,C1(C(=O)N(CCO)CC2CCCO2)CC(F)CN(C(=O)Cc2cc(F)cc(F)c2)C1 16624,N1(C(C=C2CCC(C)C2)=O)CCC2CN(C(c3ccc([N+](=O)[O-])[nH]3)=O)CC12 16625,S(=O)(=O)(c1ccc(C#N)c(N2Cc3ccc(C)cc3C2)c1)NC(CCC(=C)C)C 16626,Cc1c(NCCCCN2CCC2)nc[nH]c1=NCCNC(N1CCOCC1)=O 16627,N1(C(c2c(C#N)scc2)=O)CCCCC(CNC(=O)Cn2cnnn2)C1 16628,c1(CN(C2CN(C(=O)OC(C)(C)C)CCC2O)C)cc2n(n1)CCC2 16629,N1(CC(COC)O)CCC(N(C(=O)CC2CCN(c3ccccc3)C2)C)CC1 16630,C1(C(N2CCC(CNC(=O)CCc3cn[nH]c3)(CO)C2)=O)CCOC(=O)CC1 16631,C#CC1CCN(C(=O)C(CNC(=O)CCCOC(C)C)N(C)C)CC1 16632,c1(C(=O)NCCC2COCCN2C(C2CCCC2)=O)cc2nc[nH]c2cn1 16633,N1(C(C2CCN(C(C3(CO)CCC3)=O)C2)=O)CCCC2(CCC2)C1 16634,C1(CC)C(C(=O)NCCNC(C)=O)CCN1C(=O)CC(=O)NC 16635,CC1(C)CC(NC(c2ccc(C3CC3)cn2)=O)CN(C(c2cccnc2S)=O)C1 16636,N1(C(C(CC=C)CNC(C2C3(CC3)C23CC3)=O)=O)CCc2ccc(F)cc21 16637,N1(C(C=CCCC)=O)CC(CNC(=O)CC2C=CCC2)(OCC)C1 16638,c1(C(N2CC(COC)(CNC(C3CC3C)=O)C2)=O)noc2ccc(Cl)cc12 16639,N1(C(c2c(C)oc(CNC(=O)Cc3cc[nH]n3)n2)=O)CCc2nc(O)[nH]c2C1 16640,S(=O)(=O)(c1cc(Cl)sc1Cl)N(C(C(=O)OC)C)CCF 16641,c1(OC)cc(C)sc1C(=O)NCC1CCC1NC(c1cnc(-c2cccs2)s1)=O 16642,CC1CN(C(c2cccc(C#N)n2)=O)CCC1NC(c1cc(=O)cc[nH]1)=O 16643,C1(OC)CCC2(C(=O)NCCC(C)(C)NC(c3cccc(OC)n3)=O)CCC12 16644,C(C(C)(C(=O)N1CC(C)(CO)C1)NC(=O)Cc1ccc(C)nc1)SC 16645,c1(NC(C2(CC)CCCC2)=O)cccc(CNC(c2ccoc2Br)=O)c1 16646,C1(NC(CSCCC)=O)CCCN(C(c2c[nH]cc2C(C)(C)C)=O)CC1 16647,C1(C2(O)CCN(C(C3CC3(C)Br)=O)CC2)(NC(C=C(C)c2ccco2)=O)CC1 16648,C1(C)(CNC(c2cnc(SC)s2)=O)CN(C(C2CC23CCC3)=O)C(C)(C)C1 16649,Cc1ccc(Cl)c(CN2CCOC(CNC(c3c(O)cccc3Cl)=O)C2)c1F 16650,n1(C(C)(C)C)cc(Cl)c(=NC(=O)NCC(F)(F)F)[nH]1 16651,N1(C(c2c(OC)ccnc2O)=O)CCOCC(C)(CNC(C2(C)CCCC2)=O)C1 16652,Cc1c(C(=O)NCC(C2CC2)N(C)C(c2cc(-c3ccco3)no2)=O)nnn1C 16653,N1(Cc2ccc(OCC)cc2)CCSC2CCCCC12.c12ccc(cc1)OC2 16654,c1(CC(=O)NC2CCC(C)N(C(=O)CCCF)C2)cccc2ccsc12 16655,C1(CC(=O)OC)(NC(C2CN(Cc3ccc(C)o3)CCS2)=O)CCCCC1 16656,C1(NC(C2N(C)CCCC2)=O)C2CC3C(C2)C13C(=O)N(CC1CC1)CC1CC1 16657,c1(C(N2C3CC(CNC(C(CC#C)N(C)C)=O)C2CC3)=O)ccn2ccccc12 16658,C1(NC(C2ON=C(C)C2)=O)CCOCC1NC(c1nocc1C1CC1)=O 16659,c1(CC(=O)NCC(N(C(C(C2CCC2)OCC)=O)C)C2CC2)sc(O)nc1O 16660,C1(C(=O)NCCNC(CC2(C=C)CCC2)=O)CCN(C(=O)NC2CCCC2)CC1 16661,N1(C(CC2C(C)CCN(C(C(C)(C)OC)=O)C2)=O)CCCc2ccccc21 16662,C1(N(C)C)CCCN(CC(=O)NCCNC(=O)Cc2ccc(CO)cc2)C1 16663,CCCCN=C(NCCc1ncc(C)cn1)NCC1CC1CC 16664,CC1OCCC1CC(=O)NC(C)(C)CC=CC(=O)N(CCO)CC1CC1 16665,c1(C(=O)NCC2CCN(C(=O)Cc3cn[nH]c3)C2)cc2n(n1)CCO2 16666,C1(NC(c2nc(C(C)C)sc2)=O)CCN(C(=O)C(C)CF)C1C(C)(C)C 16667,C1(CC=CC)CCCN(C(=O)CC(C)(C)N(C(=O)C=C(C)C(C)(C)C)C)C1 16668,CCCCCC(C(=O)N1CCC(NC(c2ccn(COC)n2)=O)C1)C(C)C 16669,C1(C(=O)OCC)CCCCN1C(C1C2CN(C(C3CCCCC3)=O)CC12)=O 16670,N1(C(c2ncc(CC)cn2)=O)CCC(C2CC2)C1C(=O)N(C1CC2CCC1O2)C 16671,CC(C)(F)CC(=O)NCC1COC(CNC(c2ncsc2Br)=O)C1 16672,C(=O)(C1=NN(CCO)C(=O)CC1)N1C(CC)CN(C(c2cnc[nH]2)=O)CC1 16673,CS(=O)CCC(O)C(=O)NC12CC(NC(=O)C=Cc3cccs3)(C1)C2 16674,CCCCCC(O)C(C)C(=O)N1CC(CNC(C2Cc3nccn3C2)=O)C(O)C1 16675,c1(CC(C)NC(=O)C(Cn2cncn2)NC(c2cncs2)=O)ccccn1 16676,C=CC1CN(C(C2(N(C)C)CCCC2)=O)CC1NC(=O)CC(C)C1CCCCC1 16677,N1(C(C2C(C(=O)OC)C=C2)=O)CCCC(C(=O)NC(C2CCCCC2)C)(CC)C1 16678,c1(NC2CCSCC2)nccc(=NC2CC(NCC3CC3)C2)[nH]1 16679,C1(C(=O)NC(CC2CC2)C(=O)NCCCC2CC2)CCC(C2CC2)C1 16680,C1(CNC(CC=C)=O)CCCCC1NC(c1cnn(C2CC2(F)F)c1)=O 16681,Cc1oc(C)c(C(=O)NC2CCCC(NC(=O)CC3CC(=O)C3)C2)c1C 16682,C1(C(N2C(C)(CCC(=O)NCCC#CCO)CCC2)=O)CCCC12CCC2 16683,C1(CNC(CC(C=C)c2ccccc2)=O)CN(C(=O)C(F)(F)CC)CCCO1 16684,N1(C(C(C)c2cncs2)=O)CCCCC1CCCNC(c1ccco1)=O 16685,C1(C(=O)NC(C(N2CC(C(N)=O)OCC2)=O)c2ccco2)CC2CCCC2C1 16686,Cc1cc(=NC(C)CCNC(C2(F)CCC2)=O)c([N+](=O)[O-])c(C)[nH]1 16687,c1(C(C(=O)NCC(=C)C)NC(c2c[nH]c(C(N)=O)c2)=O)ccccc1 16688,C#CCC(C)(CC)C(=O)NCC1CC(C(=O)NCCC(C)O)=NO1 16689,N1(C(C(C)Oc2cccc(F)c2)=O)CCCC(C)(NC(C2CC(F)C2)=O)C1 16690,c1(OC)ncc(-c2cn(CC(=O)NCCc3ncc[nH]3)nn2)c(OC)n1 16691,Cc1c(C(=O)NCC(C2CCOC2)NC(=O)C2=CCCCO2)nc2sccn12 16692,C1(CC(=O)NC2C(COC)CC2)CN(C(C2CC(n3cnnc3)C2)=O)CCC1C 16693,C=CCC(C(=O)N1CCCC1CN(C(=O)Cn1ccnn1)C1CC1)C(C)(C)C 16694,c1(CN2CC(C)(CNC(c3cc(Cl)c(F)cc3F)=O)C2)cn2ccccc2n1 16695,CCCC(C(=O)N1CC(O)CC1CC(N1CC2(CC(OC)C2)C1)=O)C(C)C 16696,CC1CN(C(c2cc(=O)cc[nH]2)=O)CC1CNC(=O)CC1(O)CC1 16697,C1(C(=O)NC(C)CCNC(=O)C(N)=O)C2CCC1(c1ccco1)C2 16698,S(=O)(=O)(c1ccc(Cl)cc1)NCCC(=O)NC(CNC(CCC(=C)Cl)=O)C(C)C 16699,CCCC(CCCNC(c1ccc(CC)nc1)=O)NC(=O)CN(C)C(C)=O 16700,C1(CNC(C(C(CC)C)O)=O)C(C2CC2)CCN1C(c1ccsc1C)=O 16701,c1(NC(C23CC(C(=O)Nc4cncc(Br)n4)(C2)C3)=O)cc(O)cc(O)c1 16702,C1(C(N2CC(N(C)C(c3csc(S)n3)=O)C(F)C2)=O)CCC2(CCC2)CC1 16703,C1(C(N2C(CC(=O)OC)CCC2)=O)CN(Cc2cnc(Cl)cn2)CCN1C 16704,CC(C)(C)C#CC(=O)NCCC1CCCN(C(C2CCC(N(C)C)CC2)=O)C1 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16722,c1(C(=O)OC)cccc(F)c1CN1CCOCC1C(=O)Nc1cccnc1I 16723,N1(C(c2c(C)csc2)=O)CCCC2C1CCCN2C(=O)Cn1nc(C)c(C)c1C 16724,Cc1cc(NC(C2CC3C=CC2N(C(=O)OC(C)(C)C)C3)=O)c(I)cc1Cl 16725,CCCC(C(F)(F)F)c1nc(-c2cc(OCCOC)ccn2)nn1CC 16726,c1(OCCOC)ccc(C(=O)NCC(C)NC(=O)Cc2ccccc2)cn1 16727,C1(NC(C(=O)NC(C)C)=O)CCS(=O)(=O)C2(C1)CC(CNC(=O)CC(C)C)C2 16728,CC1(F)COCCN(C(C2CN(C(=O)CC3=CCCC3)CC2(F)F)=O)C1 16729,C1(C)(NC(CC(=O)NCC)=O)CCCN(C(C23CCC(CC2)C3)=O)C1 16730,c1(C(N2CC(CC(CNC(C(C)CC(F)F)=O)(C)C)C2)=O)c(O)cc(Cl)cc1F 16731,N1(C(C2CC3(C(OC)CC3)C2)=O)CCC(NC(=O)C(=O)N(C)C)C12CCC2 16732,C1(NC(CS(CC)=O)=O)CC1C1CCCN(C(=O)C(CO)NC(=O)C(C)C)C1 16733,c1(C(=O)OCc2c(C(N(CCC)CCC)=O)[nH]nn2)cccc(F)c1SC 16734,C(=O)(C1=CCCOCC1)N1C(CNC(=O)CC(c2cccc(F)c2)O)C2CC2C1 16735,c1(OC)cc(Cl)c(CN2CCC3CN(c4nccc(C)n4)CC23)cc1OC 16736,C1(C(=O)OC)(C(N2CC3C(NC(C)(C)C)(C3)C2)=O)CCS(=O)(=O)C1 16737,c1(OC)nc(Cl)ccc1C(N1CCC(CNC(c2ccc(Cl)cn2)=O)(OC)C1)=O 16738,c1(C(=O)NC2C(NC(C3OCCN(CC)C3)=O)CCC2)cc(=O)c(C)c[nH]1 16739,C(=O)(CCC(=O)NN(C)C)N(C(CCNC(C(CCC)NC(N)=O)=O)C)C 16740,S(=O)(=O)(c1cccc(Br)c1F)N1CCN(C(c2ccc(OC)cc2Br)=O)C(C)C1 16741,C1(O)(C(N2CCCC(CCNC(c3c(C)n[nH]c3)=O)C2)=O)CCCC(C)CC1 16742,C(C(=O)NC(C)C)(C1=CCSC1(C)C)N(C(C)CNC(C)=O)CC 16743,CCC(CC)(CC)C(=O)NCC1CN(C(C2CCC(C)(C)O2)=O)C(C)(C)C1 16744,c1(OCC(=O)NC(c2nc(C(=O)O)cs2)C)ccc(N2CCCC2=O)cc1 16745,C1(CC)CN(C(C2CC3CCC2O3)=O)CCN1C(c1ccc(NC(N)=O)cc1)=O 16746,c1(C(=O)NC2CCN(C(C(C)OC)=O)CC2F)n[nH]c2c1CCC2C 16747,C(=O)(C(CCF)NC(c1ncccc1C)=O)NC(CCC=C)C1CC1 16748,C(CCC(=O)N(C)CCNC(C1CCCC1CC)=O)N(CCC)CCC 16749,Cc1nc(C)c(NC(C2(CO)CCN(C(c3cc(C)n(C(C)C)n3)=O)C2)=O)s1 16750,N1(C(C(CC(N)=O)O)=O)CCC(C2CCCN(C(c3cnns3)=O)CC2)CC1 16751,c1(CNC(C2C(C)(C)C2(C)C)C)ccc(Cl)cc1F 16752,CC1(C)CCC(=CC(N2CCCCC2CNC(c2n[nH]cc2[N+](=O)[O-])=O)=O)CC1 16753,c1(CCC(=O)N(C2CCN(C(C3CN(C(C)C)C3)=O)C2)CC)n[nH]c(=N)s1 16754,C12(C(=O)NCC(CN(C(Cc3cc(C)ns3)=O)C)O)CC(C)(C1)OC2(C)C 16755,c1(OC)cc(C(=O)NC(Cc2cnn(C)c2O)C(=O)N2CC(C(C)C)C2)n(C)n1 16756,C1(OC)C2CC3CN(C(c4sncc4Br)C(=O)NC4CCOC4)C1C3C2 16757,C1(NC(=NCCC=C)NCCCOC2CCC2)Cc2ccccc2C1OC 16758,c1(CCC(N2C(C3(NC(C(CSC)C)=O)CC3)CCC2)=O)csc2ccccc12 16759,C(=O)(C(CCC)NC(=O)C(C)(C)O)NCc1cn(CC#C)nc1 16760,Cc1cc(F)cc(C(=O)N(CC(C)NC(c2nc(C)n(C)c2C)=O)C)c1N 16761,CC(C)C1=NOC(C)(C(=O)NC(CNC(=O)CC2CCN(C)CC2)C(C)C)C1 16762,n1(CC)nnnc1C(c1nc(C(F)(F)F)cs1)NCCC1(C)CCCC1 16763,CCC(C)CCC(=O)N(CCC(C)NC(c1cnn(CCN(C)C)c1)=O)C 16764,c1(NC)ccc(C(N2CC3CC(NC(c4cc(C)c(C)o4)=O)C2C3)=O)cc1F 16765,N1(C(C(C)SCCCC)=O)CCN(C(=O)C=C(CC)CC)CC(CO)C1 16766,c1(CNC(C2CCC3(CCC3)CC2)=O)nc2cccnc2[nH]1 16767,C12(C(=O)NCCOCCNC(C3CCS(=O)(=O)N3)=O)CCN(CC1)CC2 16768,c1(C(N2C3CC(CNC(C(COC)COC)=O)(OC3)C2)=O)nccn2nccc12 16769,c1(C(=O)NC(CCCNC(C(CSC)C)=O)(C)C)ccc(CO)cc1F 16770,C1(C(=O)NCCOc2cccnc2Cl)CCCC12CCN(C(c1cc[nH]n1)=O)C2 16771,c1(C(N2CC3C(C(=O)NC4CCCCC4(F)F)C3C2)=O)cc(F)cc(F)c1F 16772,Cc1cnc(C(N2CC(C(=O)NC3(C)CC=CCC3)C(C(C)C)C2)=O)cn1 16773,C1(C(N2CCCC(NC(=O)CCc3ccncc3)CC2)=O)CCC2(CCC2)CO1 16774,N1(C(C2CCC(OC)CC2)=O)CCC(O)C(NC(=O)Cn2nccc2C)C1 16775,N1(C(c2c(C)cc(C)s2)C(=O)NCc2ccco2)CCSCC1(C)C 16776,c1(C(N2CCC(NC(C(COC)N(C)C)=O)C2(C)C)=O)cnc2n1CCCCC2 16777,CCCCC(O)CC(=O)Nc1ccc(NC(C2COC(=O)N2)=O)c(C)c1 16778,C1(C(=O)NCC2CN(c3nccc(-n4ccnc4)n3)CCO2)C2C3CCC(C3)C12 16779,c1(C(=O)NCC2C(NC(C3CC(C)(C)C3)=O)CCC2)c[nH]c(=O)cn1 16780,n1(CC#C)cccc1C(=O)NCC1(F)CC(NC(=O)CC(C)N2CCCC2=O)C1 16781,c1(C(N(CCCOCCNC(C2C(C=C)C2)=O)C)=O)ccc(C)nc1N 16782,c1(CC)nc(C(=O)NC(C)C(C(C)C)NC(c2ccnn2CC(F)F)=O)c(C)o1 16783,C1(NC(c2c(SCC)nccn2)=O)COC2CN(C(c3cc(OC)cs3)=O)CC12 16784,C(=O)(C(CCOCCO)NC(=O)CCC1(C)N=N1)N(CC(COCC)O)C 16785,C(C1CCCN1C(=O)CSC)=CC(=O)NCCCC#C 16786,c1(C(=O)NC2CC2C(=O)Nc2ncncc2Cl)cc(O)nc2ccccc12 16787,C(CO)(C(=O)NCC1CCCN1C(C1(CC(=O)OC(C)(C)C)CC1)=O)N(C)C 16788,c1(C(=O)NCC=CCNC(C=Cc2ccc(C)cn2)=O)c(Br)ccc(C)c1F 16789,C1(C(N(C(CNC(Cn2ccc(C)n2)=O)C)C)=O)COC2(CO)CC1C2 16790,C1(C(=O)NCC2C=CCN2C(c2cnc(C3CC3)s2)=O)C(Cl)(Cl)C12CC2 16791,c1(C(N2CCOC(CCO)C2)C(=O)NCCC)cncc(C2CC2)c1 16792,N1(C(CCC(=O)N(C)C)=O)CCCC12CCN(C(=O)CCC(F)(F)C(F)F)C2 16793,S(=O)(=O)(c1ccc(NC2CCCCCC2CO)c(F)c1)NCC(CC)OC 16794,C1(NC(C(C=C)(C)CC)=O)CC2(CCN(C(C3(C#N)CCCC3)=O)CC2)C1 16795,N1(C(C2N(C(c3cnn(C=C)c3N)=O)CC2C)=O)CCC2(COC(=O)N2)C1 16796,CC1=C(c2ccccc2)CN(C(c2ncncc2Cl)=O)CC1 16797,CN1CCC(C(=O)Nc2ccccc2OCCc2nn[nH]n2)CC1=O.OCC 16798,n1(C(C)C)cc(C(=O)NC(C)C(C)NC(c2cc(N)c(Cl)cn2)=O)c(O)nc1=O 16799,c1(CC(=O)NC(C)(C)CCNC(C2CCCC2(C)C)=O)cc(Cl)cc2c1OCC2 16800,CC1CC2(CC(C(=O)NC(c3ccccc3)CNC(c3ccnc(O)c3)=O)C2)C1 16801,C1(NC(c2cc(C(C)(C)C)n[nH]2)=O)COCCC1NC(=O)C(C1CC1)C1CC1 16802,Cc1nc2cccc(C(=O)NCC(C)N(c3ncncc3C#N)C)c2[nH]1 16803,N1(C(=O)Cc2nc(Cl)cs2)CCN(Cc2ccc(Br)c(F)c2)C2CC12 16804,N1(C(c2snnc2C)C(=O)NCCCOC)CCC(CNC(C)=O)CC1 16805,c1(C(=O)NC2CC(NC(C(COC(C)C)(C)C)=O)C2)ncn2c1CCC2 16806,C1(CC(=O)NCCC2CCCN2C(=O)CN2CSCC2=O)CCCCO1 16807,c1(C(N2CC3N(S(CC)(=O)=O)C3C2)=O)cccc(Br)c1[N+](=O)[O-] 16808,C1(C(N2CCN(C(c3n[nH]c(C)c3F)=O)CC2)=O)CCC2CCCCN12 16809,N1(C(COCCCC)=O)CC2CCN(C(C3(CCCF)CC3)=O)CCC2C1 16810,N1(C(CCC(C)C)=O)CCCCC(CNC(=O)C(c2cncnc2)C)CC1 16811,c1(CC(N2CC(NC(C3C4CC5C(C4=O)C35)=O)C(CO)C2)=O)ccc(F)cc1Cl 16812,N1(c2nnc(CC)o2)CCCC2(CN(C(=O)CC(C)O)CCO2)C1 16813,N1(C(C(C)CN(C)C)=O)CC2CC(NC(=O)CCC3CCC3)CC1C2 16814,N1(Cc2nnc(C(C)(C)C)o2)CCC2(CCN(C(c3c(F)cccc3Cl)=O)C2)C1 16815,N1(C(c2nc(OC)c(C)s2)=O)CCN(C(C2CC3CCC2O3)=O)CC(CO)C1 16816,C(=O)(C(CO)C(C)(C)C)NC(C(=O)NCC(C(=O)OC)C)C 16817,N1(C(Cc2c(C)ocn2)=O)CCCC(O)(CCNC(=O)C(O)C(F)(F)F)C1 16818,C=CC(C)CC(=O)N1CCC(O)(CN(C(=O)CNC(=O)CC(C)(C)C)C)C1 16819,C(CNC(C1(S(C)(=O)=O)CCC1)=O)(C(C)C(C)C)NC(c1nc(CC)oc1)=O 16820,c1(CC(=O)NC2CC(CNC(c3cc(F)cs3)=O)C2)nnc(O)s1 16821,C1(Nc2c(OCCOC)cc(C(N)=O)cc2)CCc2nnc(C(F)F)n2C1 16822,c1(C(N2CC(C(C)NC(C=C(C)C(C)(C)C)=O)OCC2)=O)cncc(N=[N+]=[N-])c1 16823,C1(NC(C2C(OC)CCC2)=O)CCN(Cc2ncc(C)o2)CC(C)(C)C1 16824,N1(C(COCCOC)=O)CC2CN(Cc3c(Br)ccnc3Br)C2C1 16825,C1(C(=O)NC2(CNC(c3c(C)[nH]cc3)=O)CCOCC2)CC12CCOCC2 16826,c1(NC(C23CC2CN(C(C24CC(CO)(C2)C4)=O)C3)=O)cc(C(F)(F)F)cc(Cl)n1 16827,c1(CC)ccc(C(=O)N(C)CCNC(c2ccccc2CS(C)(=O)=O)=O)cn1 16828,c1(C(c2nnnn2CCSC)Nc2cnn(CCC)c2C)cc(Br)cc(F)c1O 16829,c1(C(=O)NC2CC(O)CN(C(=O)CCc3ccnc(Cl)c3)C2)cnc2nccn2c1 16830,N(C(=NCCCC(C)(C)C)NC1CCC1)CC1C(C)COCC1 16831,C1(NC(C(=Cc2cccs2)C)=O)CC2(CCN(C(=O)Cc3ccsc3Cl)C2)C1 16832,C1(NC(c2cnn[nH]2)=O)CCN(C(c2nnc(O)cc2O)=O)C(C2CC2)C1 16833,C1(NC(c2cnc(OCC)s2)=O)CCCCN(C(=O)CC2CNC(=O)C2)C1 16834,c1(C(N2CCN(C(c3c(SC)ccs3)=O)C(CO)C2)=O)cccn2nncc12 16835,C(CCCCC(=O)NCC1(O)CC(NC(C2(C)CC(F)(F)C2)=O)C1)N(C)C 16836,O=C(N=c1[nH][nH]c2ncc(Br)cc12)Nc1onc2c1CNCC2 16837,C(=O)(C1=NOC2(CCNC2)C1)N1CC(C)N(C(=O)Cc2ccc(F)cc2)CC1 16838,C1(C(N2C(CNC(=O)CCc3cccc(Cl)c3)CC2)=O)CCc2cncn2C1 16839,N1(C(c2nn(CC)c(C)c2)=O)CC2CN(Cc3ccc(C)cc3C)C2C1 16840,N1(C(CCCC)=O)CCN(C(=O)C(CC)CC)C(c2cc(F)ccc2F)C1 16841,C1(CC(NOCCCC)=O)CCN(C(c2ncoc2C2CC2)=O)CC1 16842,C(=O)(CC(F)(F)Cl)NCCOC1CCN(C(C2CC(CC(C)(C)C)C2)=O)C1 16843,CC1CC(SCc2nc(C3CCCCC3(F)F)no2)CC(C)C1 16844,CC(CC(=O)NC1C(C)(C)CN(C(=O)C2=CCCSC2)CC1(C)C)CC(C)(C)C 16845,Cc1ccc(C(=O)O)cc1CNC(C1(C(F)(F)F)CCCCO1)=O 16846,CN1CCOC(C(=O)NCC(C2CCCC2)NC(c2cnc(N(C)C)s2)=O)C1 16847,C#CC1(C(N2CC(COC)C2(C)C)=O)CN(C(C2CCCN(CC)C2)=O)C1 16848,C(=O)(CCC(C(C)C)NC(=O)CCOCC1CCC1)NC(C(=O)OC)CO 16849,c1(C(=O)NC2CC(N(C(CCOCC#C)=O)C)C2)c(C)sc(C)c1C#N 16850,N1(C(c2ccc(OC)cn2)=O)CCC(N2CCC(CCCO)CC2)C2(CC2)C1 16851,N1(C(=O)Cc2nc[nH]n2)CCC(C2CCCN(C(c3cc(CO)ccn3)=O)C2)C1 16852,N1(C(C(C)=CC)=O)CC2CC(C1)C(CO)C2NC(=O)C(O)(CC)c1ccccc1 16853,c1(N(C(C)=O)C)ccc(CSCCNC(=O)C(C(C)C)c2ccc(F)cc2)cc1 16854,C=Cc1cnn(C)c1C(=O)NC(C)CC1CN(C(=O)C(C)(C)C(=O)OCC)C1 16855,c1(C(N2CC(O)(C(C)NC(=O)CC3(CO)CC3)C2)=O)cc2n(n1)CC(F)C2 16856,CC1CCN(C(=O)CCN2CCN(C)CC2)CCN1C(C1CC2(CCC2)CO1)=O 16857,CC(F)(C(=O)NC(CNC(=O)CSCC(=O)NC1CCCCC1)C1CC1)C(F)(F)F 16858,c1(C(=O)NCC(c2cccc(C)c2)NC(c2cnns2)=O)ncc(Cl)cc1F 16859,c1(C(=O)NC(CC(C)NC(=O)C=C(Cl)Cl)C)nccc2c1[nH]c1ccccc21 16860,C1(NC(c2scc(C)c2)=O)CCN(CCNC(C2CCS(=O)(=O)C2)=O)CC1 16861,N(C1c2ccccc2C2CC12)C(N1CCC12CCOCC2)=O 16862,C(=O)(C1=CS(=O)CCC1)NCCN(CCC)C(c1cn(C(F)F)c(C)n1)=O 16863,c1(C(N(CC(CC)NC(=O)Cn2nnc(C)n2)CC)=O)cccc(O)n1 16864,N1(C(c2nccc(C)n2)=O)CC(N(C)C(c2oc(C)cc2C)=O)C2(CC2)C1 16865,c1(OC)cc(C(=O)NCC(O)CN(C(=O)C=C2CCOCC2)C)c(OC)cc1Cl 16866,Cc1ccc(N)c(C(N2CCC(C(C)NC(C3C(C)C3C)=O)C2)=O)c1 16867,c1(C(N2CCN(C(=O)Cc3cccs3)CC2)=O)cn2ccc(Cl)cc2n1 16868,N1(CC(c2cc(C)n(C(c3ccccc3)C)c2C)=O)CCc2cc(CO)ccc21 16869,C1(C)(CC)C=C(C(=O)N2CC(C)(C(=O)NC3CN(C(C)C)CC3C)C2)C1 16870,C1(C(=O)NC(CCNC(CCOC(CC(C)C)C)=O)C)CCC2C(C1)C2(F)F 16871,c1(NC(CCC)c2ccco2)cc(C(N2CCCC2CS(C)(=O)=O)=O)ncn1 16872,Cc1cc(-c2nn[nH]n2)ccc1S(=O)(=O)NC(=O)C1CCc2scnc21 16873,N1(C(CCC)=O)CCCC1(C)C(=O)NCCN(C1CCCC1)C(C)=O 16874,C1(COC)(NC(=O)CCNC(C)=O)CCN(C(=O)CC2CCNC2=O)C1 16875,C(=O)(C1CCCc2nn[nH]c21)NC1C(NC(c2cccn2C2CC2)=O)CC1 16876,c1(C(N2CC(NC(c3cnc(C)[nH]3)=O)C(F)C2)=O)c(F)cc(C(F)(F)F)cc1F 16877,C1(C(=O)NC(c2ccc(F)cc2)COC)CC2CC2N1C(=O)CSc1cnc[nH]1 16878,c1(C(=O)NCC(C)NC(c2nc(C(C)=O)sc2)=O)cc2c(s1)CCOC2 16879,C(=O)(C(F)CC(C)(C)NC(=O)C(C)=C1CC1)N1CC(OC(=O)NC)C1 16880,c1(-c2cn(CC3CN(C(C(COC)O)=O)CC3SC)nn2)ccc2c(c1)CCO2 16881,N1(C(CN(C(=O)OC)C)=O)CC2CCN(C(c3cnc(C(N)=O)cn3)=O)C2C1 16882,O(NC(=O)C(C)(C1CC1)N(C)C(c1ccc(SC)o1)=O)CCCOC 16883,c1(COC)nc(NCc2csc(Br)n2)cc(N(C(c2ccccc2)CF)C)n1 16884,N1(C(C(C2CC2)OCC)=O)CCN(C(c2c([N+](=O)[O-])cnn2C)=O)CC(C)(F)C1 16885,CC1CC(O)CCN(C(C2CC(CNC(=O)C(O)CC(F)(F)F)C2)=O)C1 16886,c1(C(N2CC(C#C)(CO)C2)=O)nn(C)c2c1CCC2 16887,C(=O)(CCCN(C)C(=N)NCc1ccco1)N(C(=O)C(O)(C1CC1)C1CC1)C(C)(C)C 16888,S(=O)(=O)(c1ccc(N2CCC(O)C(F)C2)c(C#N)c1)NC(c1cccs1)(C)C 16889,c1(OCC)ccc(C(N2CC(CO)(NC(c3ccc(F)o3)=O)C2)=O)c(F)c1F 16890,N1(C(c2n(CC)cnn2)=O)CC(NC(c2nc(Cl)cs2)=O)CC(C)C1 16891,C(=O)(CCCCCO)NC12CC(C(N3CCCC3c3ccc(Br)cc3)=O)(C1)C2 16892,C1(N(C)C)CCCN(C(C2CC23CC(NC(c2ccc(Cl)cn2)=O)C3)=O)C1 16893,C(=O)(C(O)C(C)(C)C)N1C(C(=O)NC(C2(CC(F)F)CCC2)C)CCC1 16894,CC1CCC(O)C(NC(=O)C(C(C)(C)C)NC(=O)C=CC2CC2)C1 16895,CC1CCc2nc(C(=O)NC3CCCC3NC(=O)CC3CC=CC3)cn2C1 16896,CC1(C)C(C(=O)NC2(CNC(c3cscc3Br)=O)CCOC2)C1(C)C 16897,c1(C(=O)Nc2c(C#N)scc2)ccc(F)c2c1CCC2 16898,c1(C(=O)NCC(CC)NC(=O)C(c2cn(C)nc2C)C)cncc(NC)c1 16899,c1(CN(C(c2cscc2Br)=O)C2CC2)cccc(F)c1 16900,CCC(CCCC(=O)OCC)NC1CN(C)CC(F)(F)C1 16901,c1(CC)ccc(OCCC(=O)NCC2CCN2C(=O)CC(CC)C2CCC2)cc1 16902,c1(NC(CC(CC)NC(C2CCC(=C)CC2)=O)=O)cccc2ccccc12 16903,C1(C(N2CC(SC)C2)=O)CCN(C(C2C3CCCC23)=O)C(C)C1 16904,c1(C(N2CCCC(c3noc(CCOC)n3)C2)=O)cc(F)nc(F)c1 16905,c1(CN2CC(C(N3CC4C(C3)C4(F)F)=O)NCC2)c(Cl)ccnc1Br 16906,C1(C(=O)NCCC=C=C)CN(C(=O)Cc2ccccn2)CCN1C 16907,C(=O)(C(CC(C)C)OC)NC(C(N1C(CC)(CC)CC1)=O)CC1CC1 16908,c1(-c2nc(CC(=C=C)C)n(Cc3cccc(Br)c3)n2)ccc(F)c(C)c1 16909,C1(C(=O)NC(CC#C)CO)C2CC3C(C2NC(C2CCCC(CF)C2)=O)C13 16910,c1(C(=O)NC2CCC(NC(c3nocc3C3CC3)=O)C2)cc2ccc(F)cc2o1 16911,Cc1[nH]nc2c(C(N3CC4(CNC(=O)Cc5cc[nH]n5)CCC3C4)=O)cccc12 16912,c1(-n2cc(C(C)N(C)C(c3nn(C)nc3Br)=O)nn2)cc(F)cc(F)c1 16913,n1(CC(=O)NC(C2CCCC2)CNC(=O)C2=CCC2)nc2n(c1=O)CCCCC2 16914,C(C)(C(C)(C)C(=O)NC1COC(C(C)C)C1)NC(c1cccc(CC)n1)=O 16915,N1(C(C(C)NS(C)(=O)=O)=O)CC2CC(C)N(C(=O)Cc3ccc(F)cn3)C2C1 16916,c1(OC)ccccc1C(=O)NCC(CNC(=O)Cc1sc(C)nc1C)OC 16917,C#CC1(OCC(=O)NCC(=O)NCc2noc(C(C)C)n2)COC1 16918,n1(CCC)cc(C(=O)NC2C3CC2N(C(=O)Cn2nnnc2C(C)C)C3)c(C)n1 16919,CCC(C)CCC(=O)N1CC(C2CC2C(N2CCC(COC)C2C)=O)C1 16920,N1(C(C2(c3ccc(C)cc3)CCC2)=O)CCCCCC(NC(c2cc[nH]c2)=O)C1 16921,CC1CN(C(=O)C(C)(CO)NC(=O)CN=[N+]=[N-])CCC1O 16922,C#CCC(CC(F)F)C(=O)NC(C)CCNC(=O)C=CCN(CC)CC 16923,Cc1oc(C(=O)NCC2CCC3(CCC3)C2Nc2ccccc2)cc1S(N)(=O)=O 16924,C123COC(C1)(C2)C(=O)NCC=CCNC3=O.c1(COC)ccc(C)nc1 16925,C(=O)(C(C)C(O)CC(C)C)N1C2(C(=O)NCCn3c(CC)ncc3)CC(C1)C2 16926,C1(CC(=O)NCC(C)N(C(C(=O)N(CC)CC)=O)CC)CC=CCC1 16927,c1(CCCC(=O)OC2COCCC2=O)ccc2nc(O)[nH]c2c1 16928,C1(C(=O)NCC2CN(C(C(C)(C)c3nccs3)=O)C2)CCCC2C1C2(F)F 16929,C(=O)(CCC(=O)N1CCN(C2CCC2)CC1)NCC(CC)CC 16930,N1(C(c2c(C)nn[nH]2)=O)CCC(C(=O)NC2C(O)CC2O)=C(F)C1 16931,c1(C(N(CC(C)OC)C(C)C)=O)conc1C(C)NC(=O)C(C)NC=O 16932,C=CCC(C)(N)C(=O)NC1CC(C)CCC1C 16933,c1(C(=O)NCC(CN(C(C(CC)NC(C)=O)=O)C)C)cccc2c1OCC2 16934,c1(C(N2CC(CN(C(CN(C3CC3)CC)=O)C)C2)=O)cnn(CC)n1 16935,CC1(C)CCC(C)(C(=O)NC2CCCCN(C(C3CC(=O)OC3(C)C)=O)C2)CC1 16936,C1(C)(OCC(=O)NC(C2CCN(C(=O)CC3CCOC3)C2)C)CCOCC1 16937,C1(OC)CCCC(C(=O)NCC(C2CC2)N(C(=O)C(C)=C2CCCC2)C)C1 16938,N1(C(c2c(CCC)nco2)=O)CCCC(CN(C(=O)CC(C)C2CC2)CC)C1 16939,C1(NC(CC2CCCC(C)(C)C2)=O)CCC2(CCN(C(=O)C=C3CCC3)CC2)C1 16940,C1(OC)CN2CCCC2(C(=O)NCC(C(C)C)NC(=O)Cc2nc(C)sc2C)C1 16941,C12(C(=O)NC(CC)CN(C)C(C3CC(C)(C)C3)=O)CC1COC2(C)C 16942,C1(CNC(CCn2c(C(C)C)ncc2)=O)CC2CCCCC2N1C(=O)CC(C)O 16943,C1(F)(C(=O)NCC=CCNC(C2CN(CC)C(=O)C2)=O)CC2(CCC2)C1 16944,C1(CNC(c2nc(C)n(C3CC3)c2C)=O)CCC2(CCC2)C1NC(=O)CCF 16945,c1(C(=O)NC2CC(CNC(c3c(COC)noc3)=O)C2)ccc(C(N)=O)c(Cl)c1 16946,c1(OC)cccc(C2=NOC(C(=O)NC3CCCC(C4CC4)C3)C2)c1 16947,c1(NC(CCN(C(CCCOCC=C)=O)C)C(C)C)ncc(C)c(S(C)(=O)=O)n1 16948,C(=O)(NNc1cc(Br)ccn1)NCc1cc(C)c(C(N2CCC(C)CC2)=O)cc1 16949,C1(CNC(C2(C#C)CCC2)=O)(COC)CCCN1C(=O)C(CO)N(C)C 16950,CC1(CO)CCN(C(C2(NC(C3(C)CC=CCC3)=O)CSC2)=O)C1 16951,CC(O)CC(C)(C)CNC(c1ccccc1)c1csc(-c2cnn(C)c2)n1 16952,CC(C(=O)NCC1CCC(NC(C2C=CC=CC=C2)=O)CC1)C(F)F 16953,N1(C(C(C(C)C)SC)=O)CC2CCCC(NC(c3cn(C)c(O)n3)=O)(C2)C1 16954,C(=O)(CC=C(Cl)Cl)NCCOC(C)(C)CNC(=O)C=Cc1cn[nH]c1 16955,c1(C(=O)NCC#CCNC(C2C(C)(C)COCC2)=O)c(N)cc(F)cc1Cl 16956,C12(NC(c3cnccn3)=O)CCOCC1CN(C(c1ccc(Cl)c(Cl)c1O)=O)C2 16957,N1(C(CN(C)CC)=O)CCN(C(C2CC3C=CC2O3)=O)C(CCO)C1 16958,N1(C(c2cnc(C)[nH]2)=O)CCC2(NC(c3nccc(Cl)c3F)=O)CCCCCC12 16959,Cc1cc(C(N2CCCC(c3cn(C(CN(C)C)CO)nn3)CC2)=O)nc(O)c1 16960,C1(CNC(=O)CCc2cncnc2)CC(F)CN1C(C1OCCCO1)=O 16961,c1(NC(C(=O)NC2C3CC(N)CC2C3)=O)ccc2c(c1)CCC(=O)N2CC(F)F 16962,c1(CC)onc(C)c1CNC(=O)CCN(C(C12C=CC(CC1)C2)=O)CC 16963,C1(OC(C)(C)C)CC(NC(c2sc(Br)cc2I)=O)C1(C)C 16964,N1(C(c2cc(CCC)on2)=O)CCCC(C2(NC(=O)C(F)n3ccnc3)CC2)C1 16965,C(c1cccc(C#N)c1)=CC(N1CCN(C(COCCN(C)C)=O)C2C1C2)=O 16966,c1(SCC)ccc(NC(=O)CN(CCCOC)CCCO)cc1 16967,C(=O)(C1=NN2CCCN=C2N1)N1CCN(C(C=CC(C)C)=O)CC1C 16968,c1(C(=O)NCC(CNC(C2(CC#C)CCCCO2)=O)(C)OC)cc(=O)n(C)cn1 16969,c1(C(=O)NC(C2(C(=O)N(C3CCN(C)C3=O)CCF)CC2)C)ccccc1CC#N 16970,C(=O)(C(F)CC(CC)CC)NC(CCOCC)C(N1CCC2(C=CCO2)C1)=O 16971,C1(NC(C(CCC)(C)C)=O)CCC2CC1CN2C(c1ccc(F)cc1OC)=O 16972,c1(OCCCC)cc(CNC2COC(C)(C)C2O)ccc1OC 16973,c1(C(=O)NC2C(CNC(C(N3CCC(C)CC3)=O)=O)CC2)cccc(F)c1Cl 16974,O=C(CC(C(F)F)n1ccnc1)NCCCNC(=O)C=Cc1nc[nH]n1 16975,c1(CCC)cc(C(=O)NC(C)(C)CNC(=O)C=C(C)C(C)C)ccc1Cl 16976,c1(C(=O)NCC2C(NC(c3c(CC)nccc3)=O)C2)cc2nc[nH]c2cn1 16977,c1(C(=O)NC2CCN(C(C(COC)C)=O)CC2F)nc2ccccn2c1F 16978,CS(=O)(=O)c1ccc(Cl)c(C(N2CC3CN(C(c4ccnc(Cl)c4)=O)CC23)=O)c1 16979,C1(NC(COCP(C)(C)=O)=O)CCC2CN(CC3CCN(C(C)C)CC3)CC2C1 16980,C1(C)(C(N(C2(C(=O)NCC(C(C)O)O)CCC2)C2CC2)=O)CCN(C)CC1 16981,C(=O)(C1CCCc2nc[nH]c21)N(C(CNC(C1CC2CCC(C1)O2)=O)C1CC1)C 16982,C1(C(=O)NCCC2COCCN2C(C2CCSCC2)=O)Cc2ccccc2O1 16983,Cc1c(C(=O)N(C2CCN(C(C34CC(C(C)C)(CO3)C4)=O)C2)C)cccc1Cl 16984,N1(C(=O)OC(C)(C)C)CC2CCC(NC(c3n(CC)nc(C4CC4)c3)=O)CC2C1 16985,c1(C(=O)NC(CC)CN(C(=O)COCC(C)C)C)cc(C)nn1CCO 16986,c1(C(=O)NC2C(NC(C3(C#C)CC3)=O)CCC2)c(C)cc[nH]c1=N 16987,c1(C(N2CCC(CCNC(C(C)SC)=O)CC2)=O)ncc(Cl)cc1F 16988,C1(C(=O)NCCC(C)F)(COC)CN(C(=O)CC(C)C2CC2)C1 16989,c1(C(=O)NC2C(N(C(CC(C)C3CC3)=O)C)CCCC2)ncc2cc(Cl)ccn12 16990,N#Cc1ccccc1N(Cc1cnsn1)Cc1ccccc1.N12CCCCC1C2 16991,C(=O)(C#CC(C)(C)CNC(=O)Cc1cn(C)cn1)NC(C(=O)OC)CCF 16992,c1(C(N2CC(NC(C3CC(OC)C3)=O)C2)=O)cnoc1C1CC1 16993,C(=O)(C(C)(C)C(C)NC(=O)COc1cc(C)on1)NCCCOCC#C 16994,c1(C(=O)NCCNC(N2CCCC2c2ccncc2)=O)ccccc1Cl 16995,N1(C(CN(C(C2C(C#N)C2)=O)CC2CC2)=O)CCn2cccc2C1 16996,C(N=c1[nH]c(-c2ccccn2)ccc1OC)C1(c2c(OC)cccc2)CCCC1 16997,C1(CN(C)C(c2csc(O)n2)=O)COCCN1C(c1cc(C2CCCC2)[nH]n1)=O 16998,N1(C2(NC(=O)CC3CC(NC(=O)NC(C45CCC4C5)=O)C3)CC2)C(=O)CCC1=O 16999,C1(NC(=O)Cc2ccc(Cl)cc2Cl)CC2CC(C1)N(C(=O)C(O)C1CC1)C2 17000,c1(C(N(C2CC3CN(C(COC)=O)C2C3)C)=O)cc2c(F)cc(Cl)cc2[nH]1 17001,C1(CNC(CN2C(C)CCC2C)=O)CCN(C(c2cc3sccc3s2)=O)CC1C 17002,c1(C(N2C(C(=O)Nc3cc(Cl)cnc3Cl)CC(C)C2)=O)ccc(F)c([N+](=O)[O-])c1 17003,C#CCCCCCC(=O)NCCCCC(C)(C)NC(C1CC12CC2)=O 17004,c1(NC)ccc(F)cc1C(N1CC(C(F)(F)F)OCC1CNC(=O)CCF)=O 17005,c1(C(N(C)CC2CCCC(NC(CN(C(C)C)C)=O)C2)=O)ccc(CO)c(F)c1 17006,N1(C(c2c(C)[nH]nc2CO)=O)CC2(C1)CN(C(C1COCCN1C=O)=O)C2 17007,C(=O)(CCC1=NNC(=O)CC1)N1CCN(C(C(C)N(C)C)=O)CC1CC(C)(C)C 17008,C1(CC(=O)NCCN(C(C)C)C(c2n[nH]cc2Cl)=O)CCC2(CCOCC2)CO1 17009,c1(OCC(=O)N(CC(O)CNC(C23CCCC2C3)=O)CC)ccc(C(N)=O)cc1 17010,C1(C(=O)NC2CC3CNCC23)CC2(CCCCC2)CN1 17011,c1(NCC2(NC(C3CCNC3=O)=O)C(C)CCCC2)ncc2c(n1)CCOC2 17012,c1(C(=O)NCC2CC(C)N(C(=O)CC3CCCCC3)C2)sc2nccnc2c1N 17013,CC(C)(C)C(C)(C)C(=O)N1CCOC(C(N2C3CCCC2COC3)=O)CC1 17014,N1(C(C2CC(SC)C2)=O)CC(C)CCC1CNC(c1[nH]cnc1C)=O 17015,C1(NC(c2ccc(C)c(C(F)(F)F)c2)=O)CC2CCC(C1)N2C(C1CC1(C)C)=O 17016,C(CC1CCC1)(C(=O)NC1COCC1NC(=O)C(C)Cc1ccncc1)OC 17017,c1(C(N2CC(NC(=O)C(C)(F)F)CC(C)C2)=O)cc2c(Br)cccc2c(=O)o1 17018,c1(NC(C(C)(C2CCC2)NC(=O)C(C2CCOCC2)F)=O)ccc(F)cc1 17019,C1(NC(=O)C=CC2CC2)CCC1C(=O)NCCc1cnc[nH]1 17020,c1(OC(C)C(=O)NCC2COCCN2C(c2ccc(=N)[nH]n2)=O)cccc(F)c1 17021,Cc1ccc(S(=O)(=O)N(C2CCNCC23CC3)Cc2ccsc2)cc1[N+](=O)[O-] 17022,c1(OC(C)(C)C)ccc(C(=O)OCCNC(COCCOCC)=O)cn1 17023,C1(CNC(c2ccc(F)cn2)=O)CCCC2(CN(C(=O)CCC(F)(F)F)C2)O1 17024,C1(C(=O)NC(C2CN(C(CC3CC(C)C3)=O)C2)C)NC(=O)OC1C 17025,C(=O)(CC(C)CC(C)C)NC1C(CC(=O)NC(CCCCC)C)CCC1 17026,C(=O)(C(CCC1CC1)NC(=O)Cc1cnsc1)NC(c1nc[nH]n1)CC 17027,Cc1ncccc1CC(N1CCC(NC(=O)CN(CC(C)(C)C)C)CC1)=O 17028,c1(C(C(=O)NCC(CNC(C2CCC(C)C2)=O)O)(F)F)ccc(F)cc1 17029,C1(C)(C(=O)NCCN(C(CC2CC(=C)C2)=O)CCC)CCOCC1 17030,C12(CNC(c3cn(C)nn3)=O)CCC(CN(C(C34CCC(CC3)CC4)=O)C1)C2 17031,C12(C(N(C(C(N3CC(C(=O)NCC)C3)=O)C3CC3)C)=O)CC1CNC2=O 17032,Cc1coc(C2CN(C(=O)OC(C)(C)C)C2)c1C(C)(C)C.c12cn(nn1)CC2 17033,c1(NC(C2C(NC(CS(C)(=O)=O)=O)CCC2)=O)c(Cl)ccc(F)c1F 17034,C1(SC)CC(C(=O)NCCN(C(=O)Cc2ccsc2)C(C)C)C1 17035,c1(C(=O)NCC2N(C(C3COC(=O)O3)=O)CCC2)cn(C(F)F)nc1C(F)F 17036,C1(NC(COCCN(C)C)=O)CCCC12CCN(C(c1ccc([N+](=O)[O-])o1)=O)C2 17037,C1(CN(CC(=O)NC(c2ccccc2)CC)C)(OC)CCOCC1 17038,C1(CNC(C(C)(C)C)=O)CN(C(=O)CC2C=CCC2)CCC12CCOCC2 17039,CC(C)C(N=[N+]=[N-])C(=O)N1C(C(=O)N(CC(=O)NC2CC2)C)CCC1C(C)C 17040,C(=O)(C#CC1(C)COC1)N1CC(N(C(CC(C=C)CC)=O)C)C1 17041,c1(C(=O)NC(C(C)C)C(=O)NCC2CC(C)(C)CCO2)cncc(C#N)c1 17042,C1(CNC(CSC)=O)CN(C(c2cc(C(C)(C)C)n(C)n2)=O)CC1C 17043,CCCC(O)CC(=O)NCC(CNC(c1ccc(CCC(F)(F)F)cc1)=O)CO 17044,Cc1nc(=N)[nH]cc1C(N1CCOCC(CNC(=O)Cc2ccc(F)cc2)C1)=O 17045,C#CCC(C)(C(=O)Nc1ccc(CO)c(F)c1)NC(=O)C(CC1CC1)SC 17046,N1(C(CCC=C)=O)CC2CN(c3ncncc3F)CC2C1 17047,c1(OC)cccc(C)c1NC(=O)CCCCCNC(C1NC(=O)OC1C)=O 17048,N1(C(c2c(C)cc(C)[nH]2)=O)CCN(C(=O)CCc2ncc[nH]2)CC12CC2 17049,N1(C(c2c(C)ocn2)=O)CCC2(CC1)COC(CNC(C1(C(N)=O)CCC1)=O)C2 17050,c1(C(=O)NC(C(C)NC(=O)Cn2cnnn2)C)cncc(Br)c1 17051,CC1N(C(C2CCCN(C(c3n[nH]c(C(F)(F)F)n3)=O)CC2)=O)CCC1(C)C 17052,N1(C(c2ccncc2Cl)=O)CCN(C(=O)C=CCN2CCOCC2)C2CC12 17053,C1(C(=O)NC(CCCNC(C(C=C)O)=O)(C)C)CN2CCN1CC2C 17054,N1(C(C2(COC)CN(C(=O)C(C)CC(F)F)C2)=O)CC(C)CCC1CO 17055,C(=O)(CCC(=O)NC(C)(C)CC(=O)NC(c1csnn1)C)NCC 17056,C12(CCNC(C3(F)CCCN(S(=O)(=O)CCCl)C3)=O)CC3CC(CC(C3)C1)C2 17057,N1(C(N2CC(n3cc(COCO)nn3)(C(=O)OC)C2)=O)CCC2OC(=O)OC2C1 17058,c1(C(N(C2CCN(C(c3n[nH]c(C)c3C)=O)C2)CC)=O)cncc2ccccc12 17059,c1(OC)cc(C(=O)NCC2CC2NC(C2(C)CC=CC2)=O)on1 17060,C1(CC)CCN(C(C23CCC(NC(C4CCCCC4)=O)(CC2)C3)=O)CCO1 17061,N1(C(c2occ(C)c2)=O)CCC(NC(C2(O)CCCCC2)=O)CC1C 17062,c1(OC)cc(C)c(C(=O)NCC2CC(O)CN2C(=O)CCC(N)=O)cc1Br 17063,c1(C(N2CC(O)(CC)C2)=O)nc2nc(C(=O)O)ccn2n1 17064,C(=O)(C(C)(C)C(=O)NCC1(F)CCCN(C(=O)CC2CC(C)(C)CCO2)C1)NC 17065,c1(C(N2C(C)CC(CNC(c3cncc(F)c3)=O)CC2)=O)nn(C)c2c1CCC2 17066,C1(C(=O)NCCC(O)CNC(c2cnccc2C)=O)(COC)CCCCC1 17067,N1(C(c2cc(CCC)oc2C)=O)CCN(C)CC1CNC(=O)CCC(C)O 17068,C(c1ccc(Cl)c(Cl)c1)=CC(N1CC2C(NC(=O)CC3CCCC3(F)F)(C2)C1)=O 17069,C1(C(=O)NC2(C(N(C)Cc3cc(C)no3)=O)CC(O)C2)CC(C)CCO1 17070,C=CC(C)CC(=O)NCCn1cc(CNC(c2cncs2)=O)nn1 17071,C1(C(=O)NC2CC(CCNC(c3cccc(C(F)F)c3)=O)C2)CC2CCCC2C1 17072,c1(CNC(c2cccc(Cl)c2)CO)cc(Cl)cc2c1CCC2 17073,N1(C(C(CC=C)C)=O)CCN(C(C2(CCCC)CCC2)=O)CC1C 17074,N1(CC(F)F)CC(N=c2nc3scnc3c(NCc3ccc(Cl)s3)[nH]2)C1 17075,C1(NC(COc2cn(C)nc2)=O)CN(C(c2cnns2)=O)CCC1O 17076,CC(C(=O)NC(C)(C)C(C)NC(c1sccc1Br)=O)C(=O)N1CCOCC1 17077,c1(C(=O)NCC(C)C(=O)NC2CC2)cc(=O)n(C)cn1 17078,c1(C(=O)NC(CNC(CCC(=C)C)=O)(C)CO)cc(S(C)(=O)=O)ccc1Cl 17079,C1(CC)CCCC(C(=O)OC)C1.N12CCC1C(=O)N1CC(C1)C2=O 17080,C(=O)(C(C(C)(C)C)NC(=O)CCc1ccc(C)nc1)NCc1cn(CC=C)nn1 17081,C(=O)(C(C)CC(C)(C)C)NC1CC(CNC(C2C(C)OCC2)=O)C1 17082,N1(C(C(CC)n2cccn2)=O)CCN(C(C2CCCN2C)=O)C(C)C1 17083,C1(c2onc(-c3n(C=C)ccn3)n2)CCCSC1 17084,C(=O)(C(F)(F)CCc1ccccc1)NCC(C1CCCC1)NC(C(C(C)C)O)=O 17085,N1(C(C(CCC)F)=O)CCN(C(c2cc(Cl)cn2C)=O)C(C(C)(C)C)C1 17086,c1(C(=O)NCC2C(NC(C3(Br)C(C)(C)C3)=O)C2)ccnc(C(F)(F)F)c1 17087,C1(N)(C(N(CCc2cccc(OC)c2)C)=O)CC2CCC1CC2 17088,c1(N2CC(CCCCNC(C3(C)C(CC)CCC3)=O)C2)ccc(C#N)nn1 17089,c1(C(=O)NCCC(CCNC(C2CC(=C)C2)=O)C)cc(Br)ccc1OC(C)C 17090,N1(C(c2cc(C(C)=O)c(C)o2)=O)CCN(C(c2cscc2C)=O)CC1CC(F)F 17091,c1(C(=O)NCC2CC(NC(C(C(CC)(C)C)OC)=O)C2)c(F)cccc1[N+](=O)[O-] 17092,c1(C(=O)Nc2n(C)nc(-c3ccc(Cl)cc3)n2)cc(Cl)ccc1Cl 17093,C#CCC(O)C(=O)N(C)CC1CN(C(=O)CC2CCCCC2)CCO1 17094,Cn1nc2c(c1C(N1CCC(NC(C3CCCOCC3)=O)C(F)C1)=O)COCC2 17095,C1(NC(c2c(OC)cc(C)cn2)=O)CCC2(CCN(C(=O)CC3(SC)CC3)C2)C1 17096,S(=O)(=O)(c1cnc(NC2CC3CCCC3C2)c(Cl)c1)NCCCCC 17097,C1(C(=O)NCC(C)NC(=O)C(C)(C)n2cc(Cl)cn2)(OC)CCCCC1 17098,N1(C(C=CC=CC)=O)CCN(C(=O)CC2CCC2(C)C)C(COCC)C1 17099,C(=O)(N=c1cc(Cl)nc(C)[nH]1)c1c(OC)nc(-c2ccc(C)nc2)cc1 17100,N1(C(c2c(O)nc(CC)c(C)c2)=O)CCC2(CCCN(C(=O)C3=CCC3)C2)C1 17101,C1(C(=O)N(CC(C)C#N)CC)(NC(COCCCC#C)=O)CCCC1 17102,c1(N2CC(NCc3n(CC)ncc3)OCC2)ncc2c(ccn2CC)n1 17103,N1(C(C(C)=CC2CC2)=O)CC(CNC(=O)C(F)OC(F)(F)F)C2(CC2)C1 17104,C1(NC(C2CCC2(F)F)=O)CC2CC1CN(C(c1cccn3nccc13)=O)C2 17105,Cc1nc(NC2CCCN(C(=O)Cn3nnnc3C(C)C)C2)cc(Cl)n1 17106,c1(C(=O)NCC(C(C)C)NC(c2c(CC)c[nH]c2)=O)ccc2c(c1)COC2 17107,c1(CN2CC(CNC(c3cc(C)c(C)s3)=O)C2)ccc(F)cc1F 17108,C(=O)(C1=C(Cl)CCC1)NCC1C(NC(c2ccn(CCC)n2)=O)C1 17109,CC(C)C(CCc1ccccc1)C(=O)N1CC2(CCCC2NC(=O)C=CCO)C1 17110,c1(N(c2cc(SC)ncn2)CC2(O)CNC2)ncnc2cc(F)ccc12 17111,C(=O)(CC(F)(F)F)Nc1c[nH]nc1C1CCOCC1.C12CCN(C1)C(=O)C1CCCN21 17112,CC1=C(C(=O)N2CCC(F)C(NC(c3cnc(C)[nH]c3=N)=O)C2)S(=O)(=O)CCO1 17113,N1(C(C2C(CC)CCC2)=O)CCN(C(C)CNC(=O)Cn2cccn2)CC1 17114,C1(CC)CCN(C(C2CC(=O)N(C)C2)=O)C(C(=O)NCc2ccc(OC)cn2)C1 17115,Cc1cc(F)ccc1NC(=O)Nc1cn(C)nc1OC(F)F 17116,C=CCC(CC(=O)NC(c1nc[nH]n1)(C)C)NC(C1CC2CC2C1)=O 17117,N1(C(CCCSC)=O)CCN(C(=O)Cc2ccc(C3CCC3)cc2)C(CCO)C1 17118,Cn1cnc(C=CC(=O)NCC2CC(=O)N(c3ccccc3)C2)c1 17119,N1(C(c2ccc(C)c(C#N)c2)=O)CC2(CCN(C(c3ccc(Cl)nc3)=O)CC2)C1 17120,Cc1ccc(SCC(=O)NC2CCC(CCNC(c3csc(C)n3)=O)C2)cc1 17121,c1(C(=O)NCC2(COC)CCN(C(C3CCO3)=O)CC2)nccc2ccn(C)c12 17122,N1(C(c2scc(CC)c2)C(=O)NCC2CCCO2)CCN(C)C(=O)C1C 17123,C#CCC(C)C(=O)NC(CNC(c1cnc(OCC(F)F)cn1)=O)CC(C)C 17124,c1(CC(N2CCCC(CNC(C3C(C(=O)OCC)C3)=O)C2)=O)ncc(F)cc1F 17125,C1(CNC(C(C2CCOCC2)C)=O)CCN(C(C2CC3(CCC3)C2)=O)CC1O 17126,C(=O)(CC(CN(C)C)CC(C)C)NC(C1(O)CN(c2cc(OCC)ncn2)C1)C 17127,C1(NC(=O)CCCCCn2cc(C3CCOC3)nn2)CCNCC12CCC2 17128,C1(CNC(C(C)(C)SC)=O)C2CCC1CN(C(c1ccnc(C)c1)=O)C2 17129,C1(C(C)C)CN(C(=O)CC2CCCCC2)CCN1C(C1CCCC(C)(C)O1)=O 17130,c1(C(N2CCCC(NC(C3C(C)C3)=O)C2)=O)cc(S(N)(=O)=O)cc(Cl)c1Cl 17131,C1(C(N2CCC(OC3CC3)C2)=O)COCCN(C(C2(O)CCCCCC2)=O)C1 17132,N1(C(C(C)CN(C)C(C2(CO)CCCC2)=O)=O)CCC(N=[N+]=[N-])C1 17133,C(=O)(CCOC1(C(COCC)O)CC1)N(C1CCCC1)CCCO 17134,c1(CC(N2CCC(COC)(NC(=O)CCC(C)SC)C2)=O)ccc(C)c(F)c1F 17135,c1(OCC(=O)NCC2(CNC(c3[nH]c(=NC)sc3)=O)CCC2)ccc(F)cc1Cl 17136,CC(C)(C)CC(C(=O)NCc1cccnn1)NC(=O)CCCC#N 17137,CCCC(C(=O)NC)NC(=O)C(CNC(c1ncsc1C)=O)N(C)C 17138,Cc1oc2ccccc2c1C(N1CCCC(CNC(C2(C)CCNC2=O)=O)C1)=O 17139,N1(C(C(C)=C2CCCC2)=O)CCC(C)(C)C1C(=O)N(CCCCCO)C 17140,c1(OC)ccc(NC(=O)CC2CN(C(c3ccc(C)[nH]3)=O)CCC2C)c(C)c1 17141,c1(NC(=O)CC2(NC(=O)C(F)CC3CCCC3)CC2)ccc(F)c(CO)c1 17142,C(c1cccc(F)c1F)=CC(=O)N(C(C)CN(C)C(C1COCC(C)(C)O1)=O)C 17143,c1(C(C(CC)NC(c2cn(C3CC3)nc2C(F)(F)F)=O)=O)ccc(Cl)cc1 17144,N1(C(=O)NCc2nc(C(CCC(=O)OC)C)sc2)CCS(=O)(=O)C2COCCC12 17145,C1(CC(=O)N(C)CC2(NC(c3nc(C(C)C)sc3)=O)CC2)CCCCC1C 17146,c1(COCC(=O)NCC2C=CCN2C(=O)CCC2CCCO2)ccccc1Cl 17147,c1(C(C)(C)NC(=O)NCC23CC(CO2)C3)ccc(O)cc1F 17148,Cc1n[nH]c(C)c1CC(=O)NCCCC1CCCN1C(=O)CCOC1CCCC1 17149,c1(NCCc2c(C)ncs2)cc(N(C)Cc2cccc(F)c2)ncn1 17150,c1(NC(=O)COC(F)F)cccc(CC(F)(F)F)c1 17151,N1(C(CN(C(COC)=O)C)=O)CC=C(CC(=O)NC(C)C(C)(C)C)CC1 17152,C1(CNC(C2CN(C)C(=O)C2)=O)CN(C(c2cccc(C3CC3)c2)=O)CCCO1 17153,c1(C(=O)NC2CN(C(CCCC=C)=O)CC2C)ccc2oc(O)nc2n1 17154,N1(C(C(C)CC(F)(F)F)=O)CC(CNC(=O)CS(C)(=O)=O)CC12CCOCC2 17155,CC1(C)CC(NC(C2CCCN2CC(F)(F)F)=O)CN1C(c1cncs1)=O 17156,C1(C(=O)NC2(C(=O)NC(CC(=O)NC)C)CSC2)CCC=CCCC1 17157,C=C(C)CCCC(=O)NCCC(O)C(=O)N(CCCN(C)C)CCC 17158,Cc1ccc(C(F)(F)C(=O)NC2CCC(NC(C3CCNC3=O)=O)C2)cc1 17159,c1(CC)cccnc1NC(=O)NC1CC(CNC(C2(N(C)C)CCC2)=O)C1(C)C 17160,CC(CC(C)NC(c1csc(=N)[nH]1)=O)NC(C1(C(F)F)CCCO1)=O 17161,CC1CN(c2nnc(C(F)F)o2)CC1NC(C1(C(F)F)CCCC1)=O 17162,Cc1cc(C(=O)NCC(C)N(C)C(C2CCN(C)C2=O)=O)cnc1C(F)F 17163,Cc1nn(C)c(OCC2CC2c2ccc(C(=O)N(C)C)cc2)c1OCC1CC1 17164,C#Cc1ccc(C(=O)N(C(CNC(c2cnn(C(C)C)n2)=O)CC)C)c(C)c1 17165,C1(CNC(C2(C)C(C)(C)C2)=O)CCN(C(=O)CCS(C)(=O)=O)CC1C1CC1 17166,CC1CCN(C(C2CCCC(O)C2)=O)C1CNC(=O)CC(O)c1ccccc1 17167,C1(CNC(C=CS(C)=O)=O)CCC2(CN(C(=O)C(F)(F)C3CCCC3)C2)O1 17168,C1(CNC(c2cn(C)nc2)=O)CCc2cc(N)ccc2O1 17169,Cc1sc(C(=O)NCCOC(C)(C)CNC(C2(F)CC=CC2)=O)cc1[N+](=O)[O-] 17170,C1(NC(CC(C)(C)N(C(CCCC=C)=O)C)=O)CCOC12CCOC2 17171,c1(OC)cc(O)c(C(N2CCC(C)(CNCc3cn[nH]c3)CC2)=O)cc1OC 17172,C1(C(=O)OC)COCC2(CCN(C3CN(C(CO)CO)CCC3O)C2)O1 17173,c1(C(=O)NC(C)(C)CCNC(c2cc(C3CC3)ccn2)=O)cc(Cl)cnc1O 17174,c1(OC)cccc(Cl)c1C(N1CC(NC(C2CC23CCC3)=O)CC(F)C1)=O 17175,c1(OC)nc(N2CCC(F)(C(=O)Nc3cccc(-c4nnco4)c3)C2)ncc1Br 17176,C1(OC)CN(C(=O)NCc2ccc(C)c(OC)c2)CCC1NC(=O)OC(C)(C)C 17177,CCC(C(=O)NCCC1(O)CCCN(C(C2CC(F)(CO)C2)=O)C1)C(C)(F)F 17178,CC1CC(NC(c2cc(CO)on2)=O)CN1C(c1cnc(-c2ccccc2)s1)=O 17179,CC(C)(C)C(CNC(=O)CC(=O)C(C)(C)C)C(=O)NCC(C)(O)CO 17180,C1(NC(=O)Cn2cc(Cl)cn2)CN(C(C2CC(CF)C2)=O)CC2(CC2)C1 17181,N1(C(c2oc(CC)c(C)c2)=O)CCCC(C)C1CCNC(C1(C)CC(C#N)C1)=O 17182,C(c1c(C)noc1C)=CC(N1CCCC1)=O.CC(c1cccs1)=CC(=O)NC 17183,c1(OC)cc(N2CCC(CNC(=O)CC(=O)N(C)C)(OC)C2)ccc1[N+](=O)[O-] 17184,CCCCCC(O)CC(=O)N1CCN(C)C(CNC(=O)Cc2ncccc2C)C1 17185,CC(C)CC(C(=O)NCC(C)(CO)NC(c1csc(Br)n1)=O)N(C)C 17186,c1(C(N2CC(NC(C(C)=C(C)C)=O)C3(C2)CC3)=O)nc2cccnn2c1Br 17187,N1(C2CN(CCNCC)C2)CCN(C(=O)C(COC)COC)CC1 17188,c1(C(=O)NCC(CCNC(C2CCCC(CF)C2)=O)OC)c(C)ccc(N)c1C 17189,C1(C(=O)NC(COC)COC)CN(C(c2cc(OC)ccn2)=O)CC1(C)C 17190,C1(NC(c2cc(C)c(F)cn2)=O)CN(C(=O)CCS(N)(=O)=O)C2CCCCC12 17191,C1(F)(CNC(=O)COC2CCCC2)CC(NC(c2occc2C2CC2)=O)C1 17192,C(=O)(CC(CC)CC)NC(CSCC)C(=O)NCc1cnnn1C 17193,CCC(CC)CC(F)C(=O)NC1(C(N2CCCN(C)CC2)=O)CC1 17194,c1(C(N2C(C(N(C)CCC3CCCC3)=O)C=CC2)=O)ccncc1F 17195,C1(C(N2CC(CC(C)(C)CNC(C3CCSC3)=O)C2)=O)CC(F)C(=O)N1 17196,N1(CC(C)(C)NC(=O)NC(c2sccc2C)CC)CCC(NC(C)=O)CC1 17197,c1(OC(=O)NC2C(C)CSC2)c(Cl)cc(Cl)cc1Cl 17198,C#CCCCCCCC(=O)NCc1ccc(C(=O)NC2(C3CC3)CCOC2)cn1 17199,N1(C(C(C)OCC2CC2)=O)CC2CCCC(NC(=O)C=C(Cl)Cl)(C2)C1 17200,c1(C(N(CC(CN(C(=O)CCC(N)=O)C)O)C)=O)cccc2occc12 17201,c1(C(N2CC3N(C(CCC(C)C)=O)C(CC3)C2)=O)cccc2c1OCC2C 17202,C(C(C)(C)CCNC(c1ccnc(O)c1)=O)NC(c1cn(CC=C)nc1)=O 17203,C(=O)(C(F)(F)C(F)(F)C(F)F)N1CCC(NC(C2OCC(C)(C)C2)=O)(CF)C1 17204,C(c1cn(CC(c2ccccc2)=O)cn1)=CC(=O)N(C(C)C(=O)N(C)C)C 17205,S(=O)(=O)(c1cccnc1N1CC2(CC(C)CO2)C1)NCC(c1ccsc1)OC 17206,c1(C(=O)OC)ccn2c(=O)c(-c3cccnc3-c3ccccc3)cnc2c1 17207,N1(C(CSC)=O)CC2CCCC(CNC(C3CC34CCCCC4)=O)C2C1 17208,CN1CCN(C(c2cc(CF)on2)=O)C(CNC(c2cnn(CC(F)F)c2)=O)C1 17209,c1(NC(C2C3CN(C(CCCN(C)C)=O)CC32)=O)ccc2ncnn2c1 17210,c1(CC(=O)NCC(C)(O)CNC(=O)CC2CCC2)ccccc1O 17211,c1(C(C(=O)NC(C)C)N(C)Cc2nc(CO)n[nH]2)cc(C#N)cs1 17212,N1(C(C2(CNC(C3CCCC(C)C3)=O)CCCCC2)=O)CC2(CCC(=O)NC2)C1 17213,c1(OC)ccccc1C(O)C(=O)NC1CCC1NC(=O)Cc1ccc(Cl)cn1 17214,C12(C(=O)NCC(C)(CO)NC(c3cc(OC)cc(Cl)c3)=O)CC=CCN1CCC2 17215,c1(C(=O)NC2CC(CNC(C3CCCCC3(F)F)=O)C2)cc2ccoc2cc1F 17216,N1(C(C2(COC)CCCO2)=O)CCCC(NC(=O)CCOCC2CC2)C1 17217,N1(C(CCC(CC)OC)=O)CC2=C(C1)CN(C(c1cccc(C(C)C)c1O)=O)C2 17218,C(C)(C)(CC(=O)NCc1ncccc1C(N1CCCC1)=O)OC 17219,c1(C(=O)NC(C)CCN(C(=O)C=CS(C)=O)C)cccc2nc(C(F)F)[nH]c12 17220,n1(C(C)(C)C)cnc(C(=O)NCC2(O)CC(CNC(=O)C(Cl)=CCl)C2)n1 17221,C(=O)(CCCC(=O)NC1CC2CC1N(C(=O)C(C)(C)C)C2)NC(C)C 17222,C1(NC(c2c(OC)scc2)=O)CCN(C(=O)CCn2cc(Cl)cn2)CC1F 17223,S(=O)(=O)(c1cccc(F)c1)N1CC(N(C(C(c2ccccc2)C)=O)C)C1 17224,N1(C(=O)NCCCCOC)CCCC(NCc2ccnc(OC)c2)C1 17225,n1(CCOC)ncc(C(=O)N(CC(C)(C)CNC(C2C3CCN2CC3)=O)C)c1C 17226,C1(COC)CN(C(=O)CC2(C)CC(F)(F)C2)CCN1C(C1CC(C)(C)CO1)=O 17227,S(=O)(=O)(c1ccc(F)c(F)c1)N1C2CCN(C(c3cc(Cl)ncn3)=O)C2CC1 17228,N1(C(C(=Cc2ccccc2)CC)=O)CCC2CCCC(C1)N2C(C1(F)CC1)=O 17229,c1(COC(C2C(=C)CN2C(=O)OC(C)(C)C)=O)cnc(F)c(C)c1 17230,c1(NC(C)=O)cccc(C(=O)NC2CCCN(C(=O)C(C)(C)C3CC3)C2)c1C 17231,C1(NC(C2(CC)CC2)=O)CCC(CNC(=O)COCC2CCCOC2)C1 17232,c1(CNC2CC(N(CC(=O)OCCO)C)C2)ccccc1C(F)(F)F 17233,Cn1nc(O)cc1C(N1CC(O)CC1CNC(c1ccoc1C(F)(F)F)=O)=O 17234,C(N=c1cc(NCCOc2cccc(Cl)c2)nc(C)[nH]1)c1ccc(OCC)cc1 17235,c1(C(=O)NC(CC(C)NC(COCC#C)=O)C)c(N)cc(OC)cc1F 17236,CC(C)CC(O)C(C)C(=O)N1C(C(=O)N(C)CC2(C)CCCO2)CC2CCCC12 17237,N1(C(C(C(C)(C)C)=O)=O)CCC=C(C(=O)Nc2cnn3cccnc23)C1 17238,Cc1c(Cl)c(C(F)(F)F)nn1CC(N1CCN(C(=O)C(C)CO)C(C2CC2)C1)=O 17239,C(C)(C)(CC(F)C(=O)N1CC2CC2C2CC12)NC(C1C(C(=O)OC)C1)=O 17240,CCCC(C)(O)C(=O)NCCCCC(C)NC(c1ccc(C)cn1)=O 17241,N1(C(c2nc(C)c(C)[nH]2)=O)CCC(C2CCNC2)C1 17242,C1(C(N(C(C)CNC(=O)C2=CCCCC2)C)=O)CCCC2(CCC2)C1 17243,N1(C(C2N(C(C)(C)C)CC2)=O)CC=CC(C(=O)NCC2CNC(=O)CO2)C1 17244,CC1=C(C(=O)N2CCC3(NC(c4cc(CC(C)C)c[nH]4)=O)CC3C2)CCCC1 17245,c1(C2(O)CN(C(c3cc(C(=O)OC)on3)=O)C2)ccc(-c2nn[nH]n2)cc1 17246,n1(CCCC)ncc(NC(=O)C=C2CCC2)c1CC1CCCS1 17247,C(=O)(Nn1c(C)nc2sc3c(c2c1=O)CCCCC3)c1[nH]c2ccc(C)cc2c1C 17248,c1(N(CC(C)C)C)nc(N2CCOCC(F)(F)C2)c2c(n1)CCC2 17249,Cc1ncccc1CC(=O)N(C(C(=O)NC1CC1c1cncs1)C1CC1)C 17250,N1(C(c2cnc(C)nc2)=O)CC2CCN(C(C3CCC(N(C)C)CC3)=O)CC2C1 17251,C(C(=O)NCC(C)(C)CCNC(c1ccc(C(C)(F)F)cc1)=O)(C(C)C)OC 17252,c1(OC)ccc(S(C)(=O)=O)cc1C(N1CCC(NCc2nc(Br)cs2)C1)=O 17253,CC(C(=O)NCC(=O)NCCCc1cn[nH]c1)N(C)C(C1CC1)C1CC1 17254,CCCC(C)(CC)C(=O)NC1CC2(C1)CN(C(=O)C(C(C)C)n1cnc(C)c1)C2 17255,c1(C(N2CC3C(C(=O)OC(C)(C)C)C3C2)C(=O)NC)ccc(C#N)cn1 17256,c1(C(C)C(=O)NCC2CC(F)(CNC(C3CC3F)=O)C2)ccc(F)cc1F 17257,CC(C)(O)C(C(=O)NCCCc1ccsc1)NC(=O)COCCCF 17258,N#Cc1cccc(NC(c2nnnn2CC(F)F)C2CC=CC2)c1 17259,c1(NC(C2(C)N(S(c3c(C)onc3)(=O)=O)CC2)=O)ccc2c(c1)C(=O)N(C)C2=O 17260,N1(CCOCC=C)CCN(C2CCN(C(C3CC34CC4)=O)C2)CC1 17261,N1(C(=O)COCCF)CC2CCN(C(c3cnc4c(c3)COC4)=O)C2C1 17262,c1(CC)ccc(F)c(C(N2CCC(NC(c3ccnc(O)c3F)=O)C(C)C2)=O)c1 17263,C1(COC)(CNC(=O)C(O)CSC)CCN(C(=O)C(C)(O)c2ccccc2)C1 17264,C(C)(C(C(=O)NCCCC1CC(C)C1)C(C)C)NC(C(C)=C(CC)C)=O 17265,C(=O)(C(F)(CNC(=O)C=C=C(C)C)C(C)C)NCC(COCC)O 17266,c1(C(N2CCC(O)C2c2ccccc2C)C(=O)NCC)ccc(C)c2c1CCC2 17267,N=c1cc(C(N2CCN(CCC(N3CCNCC3)=O)CC2)=O)cc[nH]1 17268,Nc1cc(C(=O)NCC2(CNC(=O)C(C3CCOCC3)F)CCC2)ccc1Cl 17269,C1(C)(CNC(C(CC)COC)=O)CCC(NC(c2csc(C3CC3)n2)=O)CC1 17270,c1(C(=O)NCC(CCCC)NC(c2cccs2)=O)n[nH]c2c1COCC2 17271,C(=O)(CCS(C)(=O)=O)NC(CCOC)C(=O)NC(CCO)C1CC1 17272,c1(CC)nc(N2CC(NC(c3cc(=O)c(OC)c[nH]3)=O)C(C)(C)C2)cc(C#N)n1 17273,c1(C(N2C(CC)CN(C(=O)Cc3csnn3)CC2)=O)cnc2sc(C)nc2c1 17274,C=CCCCC(C(=O)NC1CC(F)(F)C1)N(c1ccc(OC)cc1)CC(C)C 17275,N1(C(C2C(NC(c3ccncc3Cl)=O)C2)=O)CCc2c(cccc2[N+](=O)[O-])C1 17276,c1(CC)[nH]nc(-c2nc(CCCO)nn2Cc2ccc(Cl)cc2)c1Br 17277,C(CC(F)F)(C(=O)NCCCc1cccs1)NC(C1OCCN(C)C1)=O 17278,C1(c2ncc(C(=O)OCC)s2)CCCN(C(c2nc(Cl)c(CC)[nH]2)=O)C1 17279,C#Cc1ccnc(C(N2CCC(N(C)C(c3cccc(N)c3F)=O)C2)=O)c1 17280,N1(C(C2(NC(=O)CC3CCCSC3)CC2)=O)CCc2cncnc2C1 17281,C(=O)(C(C)CCCC(C)C)N1C(C(=O)NC(CCC)C2CC2)(COC)C=CC1 17282,CN1CC=CCC1CC(=O)NCCN(C(=O)C(F)(F)c1ncccn1)C1CC1 17283,C(=O)(CC(CC(N)=O)CC(C)C)NC(CN(C(c1c(C)nco1)=O)C)(C)C 17284,C(=O)(CCCCCC(C)C)NC(CCCCNC(CCC#C)=O)C 17285,N1(C(C(=C(C)C2CC2)F)=O)CC(CNC(=O)CN2CCS(=O)CC2)C(C)(C)C1 17286,C(=O)(C1=C(c2ccccc2)SCCO1)NC1CN(C(CC(C)(C)C#N)=O)C2C1C2 17287,c1(C(N2CC(NC(COCC(=C)C)=O)C(N=[N+]=[N-])C2)=O)cn2cccc(C)c2n1 17288,CC1CC(C(=O)N2CCN(C(=O)CNC(c3cccnc3)=O)CC2CCO)=NO1 17289,c1(C(C)C)ccc(F)c(C(=O)NCC2C(F)(F)C23CC3)c1 17290,N(C(=NCC(C(C)C)C(C)C)NCC1(F)CCCCC1)C(CC)C 17291,C1(O)(Cn2cc(C(CC)(C)C)nn2)CCN(C(=O)CCc2ccc(C)cc2)CC1 17292,Cc1ccc(C)c(C(=O)NCC2CC(NC(=O)C=Cc3cccs3)C23CCC3)n1 17293,c1(OCC)ccc(CNC(=O)CNC2CCC(NC(=O)CCC(C)=O)C2)cc1 17294,C(=O)(C(C(C)C1CCCC1)N1CCC(C(=O)NS(C)(=O)=O)CC1)NC(CC)C 17295,Cc1nc(SCC2(CO)CC23CCC3)nc(C)c1C(=O)NCC1CC1 17296,CCCCCC(C)(CC)C(=O)NC1CCC(NC(=O)CCc2ccn(C)c2)CC1 17297,C12(C(N(CCCCNC(C3CC(=O)CS3)=O)C)=O)CC3CC(CC1C3)C2 17298,C(C)(C)(CC(F)C(=O)Nc1ccc(Cl)c(O)c1)NC(c1cc(C)nnc1)=O 17299,Cn1c(O)nc2ccc(C(=O)NCCC3CCN(C(C4(C)CC4(Cl)Cl)=O)C3)cc12 17300,C=Cc1cnn(C)c1C(=O)NCC(CCCC)NC(c1scnc1CC)=O 17301,c1(CC)cnn2ccc(C(=O)NC(C)CCCNC(=O)CN(C)CC)nc12 17302,C1(CC=C)(NC(C2CC(C)(NC(=O)C=CCO)C2)=O)CCCC1 17303,C1(NC(CCC)=O)C(C)CN(C(=O)CCc2c(C)nc(N(C)C)nc2O)CC1C 17304,C(CCN(C)C(C1CC2(C1)CC(F)C2)=O)(C(C)(C)C)NC(CC(=O)OCC)=O 17305,c1(CC(C(=O)NC)NC(c2cc(F)c(C)cc2N)=O)c[nH]c2ccccc12 17306,CC1=C(Br)CCN(C(c2coc(Br)n2)C(=O)NC2CCCCC2)C1 17307,CC(C)(CCC(=O)N1CC2CC1CS2=O)NC(c1cc[nH]c(=N)n1)=O 17308,C1(=CC(=O)Nc2cnn(C)c2C(F)F)C2CC3CC(C2)CC1C3 17309,Cc1sc(C(C)N)nc1-c1nc(-c2ccccn2)nn1C 17310,c1(C(=O)NCc2nnc(CC)s2)ccc(CNC(c2oc(C)cc2C)=O)nc1 17311,N1(C(C2CC(C)OC2)=O)CCC(NC(=O)CCc2ccn(C)n2)C12CCCC2 17312,c1(CNCCN(CC)CC)nc2ccccc2n1-c1ccc(Cl)cc1 17313,CCC(CC)CC(F)C(=O)N1CCCC1C(C)(C)CNC(c1n[nH]cc1C)=O 17314,CC(C)C(C(=O)NC(C1CCCC1)CNC(=O)C(c1ccccc1)F)NC(N)=O 17315,c1(OCc2ncc(C)o2)nc(-c2cscn2)nn1CCc1csc(Cl)c1 17316,CCC(C)C(C(=O)NCC1(CNC(=O)C(C2CC(F)(F)C2)O)CC12CCC2)OC 17317,N1(C(C(CC)N(C(C(CCC)OCC)=O)C)=O)CC2CCC(C1)N2CC 17318,C1(CNC(C(CC)(C)CO)=O)N(C(c2nc(C)ccc2F)=O)CCCC1(C)C 17319,CC(F)(F)C(C)(C)CC(=O)N1CCCCCC(S(C)(=O)=O)C1.c12nccc(n1)N2 17320,C=C1CC(C)(NC(C2(OC)CCSC2)=O)C1.C12CC(C1)N(C)C2=O 17321,C1(C)(C(=O)NCc2cccc(NC(CCCCCOC)=O)c2)CC(C)OC(C)C1 17322,CC(C)C(O)C(=O)N1CC=CC1(C)C(=O)N(C)CCC1CN(C)C1 17323,C(=O)(C(C#N)C(C)(C)C)N1CC(OCCC(=O)NCc2ccc(C)cc2F)C1 17324,C12(CCNC(C(CC)(F)F)=O)CCC1CN(C(c1cncc(C)n1)=O)C2 17325,C1(C2CC2)(CNC(=O)CCc2cnoc2)CCN(C(c2cccnn2)=O)C1 17326,c1(C(C)=O)cn(CC(=O)NCCN(C(=O)CCOCC2CCCO2)C2CC2)nn1 17327,CC(C)(C)CCCC(=O)N1CCCC(CNC(C2COC(=O)C2)=O)C1 17328,CCC(Cc1ccccc1)(CCn1cc(C2(C)CCCO2)nn1)C(=O)O 17329,c1(C(C)NC(c2c(CNC(CCCOCC=C)=O)noc2)=O)cccnc1F 17330,C(=O)(C(CCOCCO)NC(=O)C(C)OC1CCCC1)N(C)CC1CC(=C)C1 17331,c1(N(CCCC(=O)NCCCN(C(C)=O)CC)CC)ccc(OC(C)C)nc1Cl 17332,C1(C(N2CCC(O)(COC)CC2)=O)CCC2(CN(C(=O)CCC(C)C)C2)O1 17333,C1(CNC(CN(C)CC)=O)CCC(NC(=O)CCc2ccccn2)CC1 17334,c1(CCC)cc(=NCCN(C)C2CC2)[nH]c(N2CCCC2)n1 17335,c1(C(N(CCNC(=O)C(c2sccc2C)=O)CC)=O)ccc(F)c(F)c1F 17336,C(=O)(C1=NN(C)C(=O)CC1)NCC(CCOC)NC(c1c(C)cccc1Cl)=O 17337,c1(N(CC(CN(C)C(C2(F)CCCCC2)=O)O)C)nc2c(cc1C#N)CCOC2 17338,Cc1cc(C(N2CC(NC(c3cc(C#N)c[nH]3)=O)C(C)(C)C2)=O)cc(Br)c1C 17339,n1(C(C)C)ncc(C(=O)NC(CNC(=O)Cn2cccn2)C(C)C)c1F 17340,C1(C(=O)NCC2(C3CC3)CCC2)(OC)CCN(C(=O)Cc2ccoc2C)C1 17341,C(=O)(C1=CC2CCC(C1)C2)N1CC2C(CN(c3ccccc3)C(C)C)(CC2)C1 17342,N1(C(C2CC(OC)CN2C(=O)CC2CCN(C)CC2)=O)CCC2(CNC(=O)O2)C1 17343,c1(C(=O)NCC(=C)CCNC(=O)CN(C)C)cnc(OC)cc1C 17344,C1(NC(Cn2cc(CN3C(C(=O)OCC)C(C)(C)C3)nn2)=O)CCC=CCCC1 17345,C12(C(=O)NCC3CC(O)(CNC(C(C)n4cccn4)=O)C3)C(=O)C3CC1C2C3 17346,c1(C(N(C)CC2N(C(C3C(C(=O)OC)CCC3)=O)CCC2)=O)cc(OC)n(C)n1 17347,c1(C(N(CCCC)CC(N)=O)=O)ccc(CNC(C2CCCS2)=O)nc1 17348,N1(C(C(C)COc2ccccc2)=O)CCCN(C(C2CCC(=O)O2)=O)CC1 17349,C=Cc1cncc(C(N2CCC3CC23C(=O)NCCc2cc(C)no2)=O)c1 17350,C1(NC(COCCSC)=O)CCN(c2ccnc(NC3CCCCC3C)n2)CC1 17351,C(=O)(CC(C)(C)COC)NC1(CC=C)CCN(C(c2cc(Br)n[nH]2)=O)C1 17352,c1(C(N2CCCC(N(C(=O)CCN3CCOCC3)C)C2)=O)ccc2c(n1)COCC2 17353,C1(CC)CC(C(N2CCC(=O)NC2=O)=O)CCN1C(C1CCCN(C)C1)=O 17354,C1(NC(C2(CCC=C)CCCC2)=O)CCN(C(C23CC(F)(C2)C3)=O)C(C)C1 17355,c1(-c2onc(-c3c(OC)cc(Cl)cc3Br)n2)cc2c(cc1Br)C(C)(C)CC2(C)C 17356,C1(NC(C(CSC)(C)C)=O)CN(C(c2cc(Cl)c(Br)[nH]2)=O)CCC1C 17357,C1(CC(C)C)CCN(C(=O)C(C(C)C)c2nn[nH]n2)CC1 17358,N1(C(C2(COCC)CCC2)=O)CCC(CN(C(=O)C(C)=C(C)C)C)CC1 17359,C1(N(C(=O)Cc2cccs2)CC)CP(C)(=O)CC1O 17360,N1(C(CCC)=O)CC(NC(c2ccc(Br)c(C)c2F)=O)C2(CCC2)C1 17361,c1(C(=O)NCc2c(CCNC(c3c[nH]nc3F)=O)ocn2)c(Cl)cccc1Cl 17362,N1(C(Cn2nc(C)oc2=O)=O)CCC(NC(C2(CO)CCCO2)=O)C(C)(C)C1 17363,c1(OCC)ccc(=NC(=O)C2CCCC(NCc3ccc4ccn(C)c4c3)C2)[nH]n1 17364,CC(C)(C)CC(C)(C)C(=O)NCC(F)CNC(c1nccnc1N)=O 17365,c1(C(=O)NC(CNC(c2nc(C)[nH]n2)=O)C)coc(=O)c2ccccc12 17366,c1(C(=O)NCC2CCC(NC(C3CC(N4CC(O)C4)C3)=O)C2)sc(F)cc1Cl 17367,c1(SC)cc(C(=O)NCC2CC2NC(=O)CS(=O)(=O)NC(C)(C)C)c(C)o1 17368,c1(OC)cc(Br)ccc1C(=O)CN(C1CCCCC1NC(=O)OC(C)(C)C)C 17369,C1(NC(c2c(C(C)(C)C)ncs2)=O)CC2CCCCCCC12 17370,n1(C(C)C)ncc(Cl)c1C(=O)NCC(C1CC1)N(C)C(C1CC1F)=O 17371,N1(C(c2cccc(-c3cn[nH]c3)c2)C(=O)NCC=C)CCC(C)C(C)(C)C1 17372,c1(C(N2CC(N(C(=O)C3=NOCC3)C)C(F)C2)=O)ccc(O)nc1Cl 17373,C1(CNC(c2cc(C3CCC3)[nH]n2)=O)CN(C(=O)CC2CCC2)CCCO1 17374,C1(NC(c2nc(CC)oc2)=O)(COC)CCN(C(c2ccc(CC3CC3)s2)=O)C1 17375,CCCCCCCC(=O)N1CC(NC(c2cc(F)ccc2C)=O)C(O)C1 17376,c1(CC)cccnc1C(=O)N(C(CC)C(=O)NC1CCN(CCF)C1)C 17377,c1(CNC(C(=O)NC(COCCOC(C)(C)C)(C)C)=O)cnn2c1CCC2 17378,Cc1sc(Cl)c(C(=O)NCCOCCCNC(=O)CCC2CCN(C)CC2)c1C 17379,CC#CCCCC(=O)N1CCCC1CCCNC(=O)COc1cccc(C)c1 17380,N1(C(C(COCC)C)=O)CCC2C1CCCN2C(c1cccc2ncnn12)=O 17381,C1(C(=O)NCC2CN(C(=O)Cc3ccsc3Cl)C2)COCCC1(F)F 17382,C1(C(N2CCN(C(=O)OC)CC2)=O)CC12CCN(Cc1ccc(I)c(O)c1)C2 17383,C1(C(N(C)Cc2c(C)cco2)=O)CC(NC(=O)Cc2cncn2C)C1(C)C 17384,N1(Cc2n(CCC(=O)OC)nnn2)CCc2c(OC(C)=O)cccc2C1 17385,c1(OC)ccc(C(=O)NC2CN(C(=O)CN3CC4CC4C3)CC23CC3)cc1OC 17386,CC1CCCC(NC(=O)Cc2csc(CNC(=O)CCn3cccn3)n2)CC1 17387,N1(Cc2c(C(=O)OCC)ccs2)CCN(C(=O)C(O)CC(C)C)C2CC12 17388,C1(NC(CCn2ncn(C)c2=O)=O)CC(NC(C2(S(C)(=O)=O)CC2)=O)C12CCC2 17389,N1(C(C(C2CCN(C(c3ccc(=N)[nH]c3)=O)C2)F)=O)CCC2=C(CCCC2)C1 17390,C#CCCCCC(=O)NCc1ncoc1CCN1CCC(n2ccnn2)C1 17391,c1(C(N2CCN(C3CN(C(C4ON=C(C)C4)=O)C3)CC2)=O)ccc(O)nc1C 17392,C1(C(=O)NC(C(C)NC(c2cc3occc3s2)=O)(C)C)CCc2nncn2C1 17393,c1(NC(N(CCN(C2CCC(F)C2)C(C)=O)CCOCCO)=O)cc(O)ccc1N 17394,C=CCC(C)(C)CC(=O)NC1CN(C(c2cnc(CC)s2)=O)CCC1CO 17395,c1(C(N2CCC(NC(c3c(CC)ocn3)=O)C2C2CC2)=O)c(F)cc(F)cc1Cl 17396,N(C1CCc2c(Br)cccc21)C(C(CC)CC)c1nnnn1Cc1ccccc1 17397,CCCC(CCC)C(=O)NCCC(C)NC(C1CCS1(=O)=O)=O 17398,C1(C(N2CCC(OCCNC(c3ccc(SC)cc3)=O)C2)=O)CCCCN1N=O 17399,c1(C(=O)NCC2(CCNC(CN(C3CC3)CC)=O)CC2)cc(C(N)=O)co1 17400,C=C(C)CCCNC(=O)COC(C)(C)CNC(=O)C(=O)NCC(F)(F)F 17401,O=C(C1=C(F)CN(C(C2(F)CCOC2)=O)CC1)NCc1nn[nH]n1 17402,c1(C(N(C(C(N2CCC(NC(=O)NC)C2)=O)C)C)=O)nn(C)cc1C 17403,N1(C(CNC=O)=O)CCOCC1CCNC(=O)COC1CCOC1 17404,O=C1COC(C(=O)NCCCNC(=O)Cc2cnn(Cc3ccccc3)c2)C1 17405,c1(C(=O)NCC(C)(C)NC(=O)Cc2ccc3c(c2)CCC3)cc(Cl)c([N+](=O)[O-])[nH]1 17406,N1(C(CCS(C)=O)=O)CCC(NC(=O)Cc2ccc(F)c(Cl)c2)C12CC2 17407,c1(C(N(CC(CNC(Cc2scc(C)n2)=O)C)C)=O)cccc(C2CC2)n1 17408,CCCC(O)(CCC)CC(=O)N1CCCC(C2(NC(C3(N(C)C)CC3)=O)CC2)C1 17409,C(c1cnn(C)c1C)=CC(N1CC=CC(NC(c2ccc(NC)cc2)=O)C1)=O 17410,c1(NC(C2(NC(=O)OC(C)(C)C)CC23CCC3)=O)cnnc2ccccc12 17411,c1(-c2cnc(SCC(=O)OCC(=O)Nc3cnn(C)n3)o2)cccc(F)c1 17412,C(=O)(C1CCCc2nncn21)N(CCN(C(=O)C=Cc1ccco1)C)C 17413,S(=O)(=O)(c1ccc(C(N2CCC(C)(CNC(c3ccoc3)=O)C2)=O)cc1)NCC 17414,c1(C(=O)NCC(CC=C)NC(c2nn(C)nc2Br)=O)cnc(C)n1C 17415,N1(C(c2cc(CCC)on2)=O)CCCC(CC(=O)NC2CC3CCC2O3)C1 17416,CC1CN(C(=O)C=C(Cl)Cl)CC2(CCN(C(c3ccc(S(N)(=O)=O)o3)=O)C2)O1 17417,c1(CSC)c(C(=O)NC(C2CN(C(c3csc(=N)[nH]3)=O)C2)C)oc2ccccc12 17418,C1(NC(C(C)(C)OC)=O)C2CN(C(C3CCCC3C(C)C)=O)CC12 17419,C1(C)(NC(c2ncn(C(C)C)n2)=O)CCN(C(c2cc3n(n2)CCO3)=O)CC1 17420,c1(C(=O)NC2C=CCN(C(CCOCCC)=O)C2)c(C)[nH]c2ccc(F)cc12 17421,N1(C(c2c(C)csc2C)=O)CCCN(C(=O)C=CCCc2ccccc2)CC1 17422,S(=O)(=O)(c1csc(C(N2CC(CNC(=O)C(C)(C)F)C3CC23)=O)c1)NC 17423,c1(C(N2CCC(CC=C)(NC(=O)C=C(C)C(F)F)C2)=O)cnc2ccc(F)cc2c1 17424,c1(C(N2CC3C(CNC(c4n(CC)cnn4)=O)(C3)C2)=O)ccc2c(n1)CCCC2 17425,CC(O)CC(=O)NC(Cc1cc[nH]n1)C(=O)N1CC(O)(c2cc[nH]n2)C1 17426,CN1C(=O)Cc2ccc(-c3cccc(CN4CCC(CC#N)CC4)c3)cc21 17427,N#Cc1cc(N2CCC(NC(=O)CSc3n[nH]c(O)n3)C2)nc(C2CC2)n1 17428,C1(NC(c2c(CC)occ2C)=O)CN(C(c2oncc2C)=O)CCC1F 17429,CC1CCCN(C(c2cnsc2)=O)C1CNC(C1OCCN(C)C1=O)=O 17430,C1(C(N(CC(C2CC2)OC)C)=O)CN(C(c2cn(C)cc2C)=O)CC1(F)F 17431,c1(NCC=CCNC(CC2C(OC)COCC2)=O)ncn(C)c(=O)c1Br 17432,c1(C(=O)NCCCCCN(C(C)C)C(C2CSCCS2)=O)ccc(O)c(F)c1F 17433,C=CCCCCC(=O)N1CC(C)C(C)(CNC(C2CCCS2)=O)C1 17434,c1(C(C2CC2)NC(=O)NC(CC)CCCO)cc(Cl)ccc1Cl 17435,CC1(C)CC(NC(C2CC2c2ccc(Cl)cc2)=O)CN1C(c1ccc(F)cn1)=O 17436,C(CCCC(=O)NC(C)(C)C(=O)N1CCC1C(C)C)OC 17437,C1(N2CC(C(=O)OC(C)(C)C)CC(OC)C2)CC2CCC1C1C(=O)NC(=O)C21 17438,C1(C(=O)OCC(=O)Nc2c(C)cc(C)nc2)CCc2nnc(O)n2C1 17439,c1(C(N2CCN(C(C3CC3c3ccccc3)=O)C3C2C3)=O)cn2ncccc2n1 17440,N(C1CC(F)(F)c2ccccc21)C(=O)C(N1CCc2ccc(F)cc21)=O 17441,Cc1nc2cc(C(=O)NCC3(F)CCN(C(c4cnc[nH]c4=N)=O)C3)[nH]c2s1 17442,CCC(CCCC(=O)NCc1csc(C)c1)NC(=O)C(C)OCCOC 17443,C1(CC(N2CCC(COC)(NC(=O)C3=COCC3)CC2)=O)CC(C)CC(C)(C)C1 17444,c1(CC)cc(C(N2CCOC(c3cccs3)C2)C(=O)NCC(C)C)n(C)n1 17445,c1(C(=O)NC2CC(C(N(CCCC(C)O)C)=O)C23CCC3)cccc2[nH]ncc12 17446,Cc1c(NC(=O)C(=O)N(C)CCC2CCCN2C)cnn1-c1ccncc1 17447,CCC(CC)C(C)C(=O)N1CCN(C(=O)CC(F)(F)CC)C(c2ccccc2)C1 17448,C=CC1COCCN1C(=O)C(C)(C)NC(=O)CC1CC1C1CC1 17449,CC1CCC(CCC(=O)N(C(Cc2ccco2)CO)C(C)C)O1 17450,c1(CN2CCCC(CN(C)C(c3cccnc3S)=O)C2)cccc2ncccc12 17451,C(=O)(CCCC(C)(C)C(=O)OCC)NC(C(C)NC(CSCCC)=O)C(C)C 17452,Cc1ccc(CNC(C2C3CC3CN2C(=O)CCC2CC2C)=O)nn1 17453,N1(C(C2(S(N)(=O)=O)CC2)=O)CC2CCCC(C1)N2C(=O)CCn1cccn1 17454,c1(C(N(C2CCCCCC2)CCNC(c2c(C)n[nH]c2)=O)=O)nnn2c1CCCC2 17455,c1(C(N2CC(NC(CS(=O)(=O)NC)=O)C(F)CC2)=O)ccc2c(c1)OCCCO2 17456,N1(Cc2ccc(C#C)s2)CCN(C(c2cc(F)c(Cl)cc2F)=O)C(C#N)C1 17457,Cc1cc(C(=O)NC2CN(C(=O)C(O)Cc3cnc[nH]3)CC2(C)C)c(N)c(Cl)c1 17458,C1(NC(c2cnn(CC)n2)=O)CC2(C(=O)NCC3CC(=O)N(C)C3=O)COC1C2 17459,c1(C(N(C2CN(C(=O)CN3CCNC(=O)C3)CC2O)C)=O)cc2occc2n1C 17460,C(C(=O)N(CC(C)(C)NC(=O)C(O)C(F)F)C)(C(C)C)NC(CC(C)C)=O 17461,N1(C(C=CC(CC)=CC)=O)CC2CCN(C(c3scc(C)c3Cl)=O)C2C1 17462,Cn1cnc2c(C(N3CCOC(CNC(=O)CC4(C)CCCO4)C3)=O)ccnc12 17463,Cc1cc(C(N2CC(C)C(C)(CNC(=O)CSC(C)C)C2)=O)nnc1C 17464,CCCCCC(CC)C(=O)NC1CCC1CNC(c1cnnc(C)c1)=O 17465,C(c1ccc(F)c(F)c1)=C(CCC(=O)N(c1ccc(F)cc1C)CC)C 17466,c1(CC)nn(C)cc1C(=O)NC(C)(C)C(C)NC(=O)CCc1cn(C)nc1C 17467,Cc1cc(C)c(S(=O)(=O)N2CCC(O)(CC(=O)N(CC(O)CO)C)CC2)c(C)c1 17468,O=C1CSC(C(N2CCCC2CCNC(c2ccncn2)=O)=O)C1 17469,N1(C(c2cc(C(C)C)on2)=O)CCCC(C(C)C(=O)NC2CCN(C3CC3)C2)C1 17470,C1(C)(NC(C)=O)CCN(C(c2sc(C(C)(C)C)nc2C)=O)C1 17471,C1(C(N(CC(NOCCC=C)=O)C(C)C)=O)CC12CCCC2 17472,C(=O)(C(C)(C)CC(F)F)N1CC(C(=O)NC(C)CC(C)(C)O)C(C)C1 17473,CCC(C(=O)N1CCC(C2CCCN2C(C2CCC(OCC)CC2)=O)C1)C(C)C 17474,Cc1sc(O)nc1C(N1CC(C(N)=O)(CNC(=O)Cn2cnnc2)C1)=O 17475,CC1OCC2(CCN(C(=O)CC3CCCN3Cc3ncc(Br)cc3F)CC2)C1N 17476,CC1C(C)CCN1C(c1c[nH]nc1CCNC(=O)CCC(=O)N(C)C)=O 17477,N1(C(C(C)(N(C(c2c(C)nc(C)o2)=O)C)C2CC2)=O)CCN(C)C(C2CC2)C1 17478,c1(OCCCN2C(NC(=O)Cc3cscn3)CC2)ccccc1C(=O)O 17479,C(CCNC(C1CC1OC(C)(C)C)=O)(C(=O)NCC(O)(CO)CO)OC 17480,CC1CN(C(C2CS(=O)C2)=O)CCC1NC(=O)CC(C)(O)C1CC1 17481,CC(C)(C)CCCCC(=O)NC1CN(C(c2ccn(C(F)F)n2)=O)CC(C)(C)C1 17482,C(C)(CCC(=O)NCC1CCCC1C(=O)NC1(CCF)CC1)OC 17483,c1(OCCCC(=O)OCC2(c3nn[nH]n3)CCCOC2)cc(Cl)c(Cl)cc1Cl 17484,C1(NC(c2sc(CC)c(C)c2)=O)CN(C(C2(CCOC)CCC2)=O)CC1(C)C 17485,CC1CC2CN1CCC2.C(=O)(CC(F)(F)F)NC(=O)CC1CC2CCC1O2 17486,c1(CC)ccc(C(=O)NCC(Cc2ccccc2)CC(=O)OC)cc1CC 17487,C1(NCCC2N(C(CCC(=O)NC3(C)CC3)=O)CCSC2)CCCC(F)(F)CC1 17488,N1(C(C=CCC)=O)CCC(NC(c2cc(C(C)=O)c[nH]2)=O)CC1 17489,C12(C(N3CCC(NC(c4[nH]cc(C)c4)=O)C3)=O)CCCC(C)(C1)OC2 17490,c1(COC)cncc(C(=O)NCCOCCCNC(=O)CC(C)n2cccc2)c1 17491,C1(CNC(c2cc(C)ns2)=O)CC(F)(F)CN1C(c1ccc(N)c(Cl)n1)=O 17492,N1(C(c2n(CC)ccc2)=O)CC(NC(c2cc(-c3ccccc3)co2)=O)C(C)C1 17493,CCCCN=C(NCC1CC2CCCC2C1)NCC(N1CCOCC1)(C)C 17494,N1(C(CSS(C)(=O)=O)=O)C2CCC1CC(NC(c1cc(Cl)no1)=O)C2 17495,C=CC(CC)CC(=O)N1CCC(N(C(c2ccnc(C(C)(F)F)c2)=O)CC)CC1 17496,CC1(C)CCC=C1C(=O)NCC12CN(C(C3SCCCS3)=O)CC1(C(F)(F)F)C2 17497,CN=c1cc(C(=O)NCC(c2cn(C(C)C)nn2)(C)C)c(Br)c[nH]1 17498,C1(CNC(C(C)SC(F)(F)F)=O)CN(C(=O)COCc2ccnn2C)CCN1C 17499,C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NCCNC(c1cc(F)c(OC)c(F)c1)=O 17500,c1(CN2CCC(N(C(c3cccc(CC)n3)=O)C)C2)ccc2c(c1)OCCO2 17501,C1(CNC(C2(NC(=O)NC)CCCC2)=O)CCC(NC(C2CC2CF)=O)CC1 17502,C=CCCC(O)CN(C)C(C1CC(F)CN1C(=O)C=C1CCCCC1)=O 17503,C1(NC(Cn2c(C)cnc2)=O)CC2CC1N(C(C1(NC(N)=O)CC1)=O)C2 17504,c1(CC)ncc(Br)cc1C(N1CCC1CNC(C1(CC2CC2)CCC1)=O)=O 17505,c1(C(N2CCC(CC(=O)Nc3ccc(CC)nc3)CC2)=O)c(OC)cccc1F 17506,c1(CCC(=O)NCCCC2(NC(C3CCC(C)S3)=O)CC2)cccc([N+](=O)[O-])c1 17507,c1(NC(C2N(C(c3cc(C(C)C)on3)=O)CC(F)C2)=O)cnc2ccc(F)cn12 17508,CC1(NC(N2CC34CCC3(COC4)C2)=O)CS(=O)(=O)CCO1 17509,Cc1ccc(C(N2CCC(C(C)(O)CNC(C3CC(O)C3)=O)CC2)=O)c(C)n1 17510,C12(CN3CCN(CC(N4CCCC4)=O)C(C)C3)COCC(C3CC3)(C1)C2 17511,CC1CCC(CCC(=O)N(C)CC2CN(C(=O)CCCC3CC3)C2)O1 17512,c1(C(N2CC(CC)N(C(c3cccc(=O)o3)=O)CC2)=O)ccc2c(c1)COCC2 17513,N1(C(Cc2cc(C)on2)=O)CCOC2CN(C(=O)C(C)(O)C(F)(F)F)CC12 17514,C12(NC(CC(C)C3CC3)=O)CCCN(C(=O)COc3ccccc3O)CC1C2 17515,N1(C(C(CO)NC(N)=O)=O)CCCC(CNC(C2(S(N)(=O)=O)CC2)=O)CC1 17516,C1(NC(C(CCC)NC(N)=O)=O)CCN(C(=O)CS(=O)(=O)CC)CCC1CO 17517,C(=O)(C1=CS(=O)CCC1)N1C(CC(=O)OC)C2CCC1C2 17518,c1(CC(N2CCC(N(C(=O)C(F)C(C)C)CCC)C2)=O)cc(F)cc([N+](=O)[O-])c1 17519,c1(C(=O)NCCCCCNC(C2(C)CC2(Cl)Cl)=O)cc2c(nn1)CCC2 17520,Cc1cc(F)c(C(=O)NCC(C)(C(C)C)NC(c2ncsc2C)=O)c(Cl)c1 17521,CC1CCN(S(=O)(=O)CCn2cncn2)CCC1N1CCC(F)C1 17522,c1(OC)ccc(-c2noc(C3CCCC3N)n2)c(Cl)c1 17523,N1(C(C2C(=O)NCC2)=O)CCC2CC1CN(C(c1ccc3c[nH]nc3c1)=O)C2 17524,c1(C(=O)NCC2N(C(C3(SC)CCC3)=O)CCCC2)noc2ncccc12 17525,Cn1cc(CC(=O)NC(c2cn(C(C)(C)C(=O)O)nn2)(C)C)cn1.C1(CO)CCC1 17526,N1(C(CONC(C(C)c2cc(C)no2)=O)=O)CC2CCCC(O)C2C1 17527,CC1(CC(=O)NCC(C2CC2)NC(=O)C(F)=C2CCC2)CC1(F)Cl 17528,N1(C(CCc2nnc(C(C)C)o2)=O)CCN(C(=O)C=CCF)CC12CCC2 17529,c1(C(N2CCC(CNC(c3cncc(OCC)c3)=O)C2)=O)ccnc([N+](=O)[O-])c1 17530,N1(C(C(C)C2(O)CCC2)=O)C(C(=O)NCCOC2CC2)CCC1C 17531,C1(O)(CC(C)C)CCN(C(=O)CC2(N(C)C(c3ccnnc3)=O)CC2)C1 17532,CC1(CNC(C2(F)CC=CCC2)=O)COCCN(C(c2ccc(Cl)c(O)c2)=O)C1 17533,c1(CC(=O)NC(CSC)(C)C(=O)N2CC(c3nc(C)no3)C2)cccc(C#N)c1 17534,C#CCC(CC#C)C(=O)NCC(C)NC(=O)CCc1cccc(OCCC)c1 17535,c1(C(N2CCN(CC(N3CCCC(C)(O)C3)=O)CC2)=O)ccc([N+](=O)[O-])cc1Br 17536,c1(NC(C(COCC)C)=O)cccc(-c2nncn2C)c1 17537,C1(NC(c2c(SC)n(C)nc2)=O)CN(C(=O)CN2CCCCC2)CC(C)(C)C1 17538,N1(C(=O)C=Cc2cscn2)CCCN(C(=O)CC2CCC3(CCC3)O2)CCC1 17539,N1(C(c2cc(C(C)(F)F)on2)=O)CC2CCN(C(C3(c4cc[nH]n4)CC3)=O)C2C1 17540,C12(NC(c3cc(C(F)F)ccn3)=O)CCC1CN(C(=O)CC1CCCCC1O)C2 17541,c1(NC(CN(CC)CC2C(NC(=O)C(C)SC3CC3)CC2)=O)ccccc1Cl 17542,C(=O)(C#CC1CCOCC1)NCC(CCC)C(=O)N(C)CCOC1CC1 17543,c1(OC)cc(OC)c2ccnc(NCc3cccnc3C)c2c1 17544,c1(C(C)C)ccc(C(=O)NCCn2cc(-c3cccs3)nn2)cc1F 17545,c1(CCC(=O)NCCN(C(=O)C(C)NCC(F)(F)F)CCOC)nccn1CC 17546,c1(C(=O)NC2C(CC(=O)NC(CCCC)C)C(O)C2)ccnc2cc[nH]c12 17547,c1(C(C)=O)ccc(C(=O)NC(C)(C)CNC(=O)C(C)OCc2ccccc2)nc1 17548,C1(C(N(C(C)C(=O)NCC(C(C)(C)C)OC)CC)=O)CCN(C)C(=O)C1 17549,c1(CC(=O)OC)ccnc(NCC2(CCNC(c3occc3Br)=O)CC2)n1 17550,C(CC(C)CCNC(c1nocc1Br)=O)NC(C(C)OC1CCCC1)=O 17551,C12(NC(CC(C)OC)=O)CCC(NC(=O)CCNc3nc(C)cs3)(C1)OC2 17552,N1(C(C(CC=CC)C)=O)CC(CNC(=O)CC2CCC2C)CC12CCC2 17553,C1(C)(C(=O)NCC(C)CN(C)C(c2cnn(C(F)(F)F)c2)=O)CCNC1 17554,C1(C(N2CCCC(CCC(=O)NC3(C)CCC3)C2)=O)CC2CCCC2C1 17555,C1(NC(C(C(CC)O)C)=O)CCN(C(=O)C(C)(O)c2ccccn2)CC12CCC2 17556,c1(C(C(=O)NC2CC(NC(c3c(CC)occ3)=O)C2)(F)F)ccc(Br)cn1 17557,c1(CC(=O)N(C)C)ccc(NC(=O)C(N2CCSCC2)=O)cc1 17558,C(=O)(C(C)(C)C(=O)NCCC(COC(c1cc(Cl)ncc1OC)=O)OC)OC 17559,CC1(C)CCCC(C(=O)NC2CN(C(c3cccnn3)=O)CC2(C)C)C1 17560,N(C(=NCCc1ncccc1C)NCc1nn(C)cc1Br)C(COC)C 17561,N1(C(C(C)n2cccn2)=O)CCN2CCN(C(=O)C(C)n3ccnc3)CC2C1 17562,N1(C(C(C)=CC2CC2)=O)C2CCCC1CN(C(C1CC3CCC1O3)=O)C2 17563,CCC(CC)C(C)C(=O)N(CC(=O)NC1(COC)CC(C)(C)C1)CCOC 17564,c1(CC)occc1C(=O)N(CCCN(C(=O)CC#N)C)C 17565,c1(C(N(CCC(N2CC(CC)C(NC(N)=O)CC2)=O)C)=O)cc(C)cc(C)c1N 17566,C12(NC(C(C)CC(C)(C)C)=O)CN(C(=O)Cn3cnnc3O)CC1CS(=O)(=O)C2 17567,CC1CCCN(C(c2cnn(C(F)(F)F)c2)=O)C1CNC(c1ccsn1)=O 17568,c1(NCC(CCC)C)ncccc1S(=O)(=O)NC1(c2cc(F)cc(F)c2)CC1 17569,C1(CNC(=O)COCC2CCOC2)CC2CCC(C1)N2C(=O)C=Cc1cnc[nH]1 17570,c1(C(=O)NCC(C2CCN(C(CC(C)SC)=O)CC2)(C)C)c(O)cccc1F 17571,CCCCC(F)C(=O)NC1CC(OCC(N2CCC(C(F)(F)F)C2)=O)C1 17572,c1(CC)cccc(C(=O)NC2CCC(CNC(=O)CC3(OCC)CCCC3)C2)n1 17573,CCC(CC(=O)N(CC(=O)NC(C)Cn1cnnc1)C1CC1)CC(C)C 17574,C1(F)(CNC(C=CCCC)=O)CCN(C(=O)CN(C)CCOC)C1 17575,C(=O)(C(O)CC(C)(C)C)NCC1(CO)CCN(C(C=CC(C)C)=O)C1 17576,C(=O)(C1=C(Cl)CCC(C)C1)NCC1(CNC(C(C)S(N)(=O)=O)=O)CCC1 17577,C1(C(=O)Nc2n(C)c(C#N)cc2)CC2(CCCCN2C(=O)COCP(C)(C)=O)C1 17578,N1(C(CCC)=O)CCCC(CCNC(=O)C(c2cc(Cl)cc(Cl)c2)(C)C)CC1 17579,Cc1ccc(CSc2ccc(C(=O)NC3(C4CCCCO4)CC3)o2)cc1 17580,c1(C(F)(F)F)cc(C(c2nnnn2C2CCC2)NCC2CCC2)on1 17581,CN1CC(=O)N(CC(=O)NCC(O)CCNC(C2(CO)CC(C)(C)C2)=O)C1=O 17582,c1(C(N2C(C)(CNC(C(C=C)(C)CC)=O)CCC2)=O)cc(S(=O)(=O)NC)oc1C 17583,C(C(=O)NOCC1CCS(=O)(=O)C1)(c1ccccc1)N.CC(C)=CCC(=O)N 17584,C=CCC(C(=O)NCCC1(SC)CN(C(=O)C(C2CCCCC2)O)C1)NC(C)=O 17585,N1(C(C2CN(C(C)=O)C2)=O)CC(N(C)C)C(CNC(=O)Cc2csc(C)n2)C1 17586,N1(C(c2nn(CC)c(C)c2)=O)CCC2(CCCN2C(=O)C(O)C2CC2)CC1 17587,Cc1nn2cc(C(=O)NC3CC(C)N(C(=O)CSCc4ccccn4)C3)nc2s1 17588,C1(C)(C(=O)NC2CCN(C(COCC#C)=O)C2C2CC2)CCS(=O)(=O)CC1 17589,CON(CCC(=O)N(C)C(c1ncccn1)C)C(=O)C1(C#N)CCOC1 17590,N1(C(CCNC(=O)NCC)=O)CC(OC)CC(NC(c2ccc(O)nc2Cl)=O)C1 17591,CC(C)CC(C)(C)CNC(C1CCN(C(=O)C2C(C)(C)C2(F)F)O1)=O 17592,C1(C(=O)NC(CC)CNC(=O)CC(O)C2CC2)CCC2CC2CC1 17593,C1(CC)C(C(=O)NCCC2C=CCC2)CCN1C(=O)CCN1CCCCC1 17594,c1(NC(C2COCCN2C(C2CC(O)C2)=O)=O)c(F)c(F)nc(F)c1F 17595,c1(C(=O)NC)cc(C)[nH]c(=NCC2CCCC2NC(c2nn(C)cc2Cl)=O)n1 17596,C1(C)(CNC(c2n(CCCC)nnn2)c2ccnn2COC)CCC(=O)N1 17597,CC1(C)C(NC(c2ccnc(C(=O)N(C)C)c2)=O)CCN1C(c1nccs1)=O 17598,c1(C(=O)NC2CCN(C(c3c(C)c(F)ccc3N)=O)C2)c(F)cccc1[N+](=O)[O-] 17599,CS(C)(=O)=NCC(=O)NC1CCOCC1NC(=O)C=Cc1ccccn1 17600,C#CCC(CC(F)F)C(=O)N1CCC(OCC(N2CC(CC(=O)OC)C2)=O)C1 17601,C12(NC(C=CS(C)=O)=O)CCOCC1CN(C(c1cccc3oncc13)=O)C2 17602,C1(CN=C(NC2C(C)C2)NCc2ccc(Cl)c(Cl)c2)CC2(CCOCC2)C1 17603,c1(C(=O)Nc2c(OCC)cccc2)ccc2[nH]nc(-c3c(C)nn(C)c3C)c2c1 17604,N1(C(CC2C(=O)NCC2)=O)CCC(C(F)F)(CNC(c2ccsn2)=O)C1 17605,c1(C(=O)NCC=CCNC(C2C(CC)CCCC2)=O)nn(C)c(N)c1C 17606,Cc1nc(SCC(=O)NC(CNC(=O)C(C)N2CCCC2)C2CCC2)n[nH]1 17607,Cc1ccc(-c2ccnn2C)cc1NC(N1CCC(c2ncc(Br)cn2)C1)=O 17608,N1(C(CCCOC(C)=O)=O)CC2CCC2(CNC(=O)CN2CCS(=O)(=O)CC2)C1 17609,C1(NC(C2C(CC(=O)OC)CC2)=O)CCCN(c2ncc[nH]c2=O)C1 17610,N1(C(C2(COC)COC2)=O)CCC12CN(C(C1CCCC3(CC3)C1)=O)C2 17611,c1(C(=O)NC(CN(C(=O)C2=CCCC2(C)C)C)(C)C)cc(F)cc(N)c1F 17612,C(=O)(CCS(C)(=O)=O)NCC(CC)(CC)NC(C1CC2C=CC1O2)=O 17613,Cc1cc(Cl)ccc1C(=O)N(CCN(C)C(C1(CO)CCCC1)=O)C1CC1 17614,C1(NC(c2n(C)ccc2)=O)CC2CC1CN(C(C1CNC(=O)CC1(C)C)=O)C2 17615,C1(NC(Cn2c(C)nnn2)=O)CN(CC(F)(F)F)CCC1c1ccccc1 17616,Cn1cc2c(n1)CCC(C(N1CCC(NC(=O)C=Cc3ccc(Cl)cc3)C1)=O)C2 17617,N(C1CCOc2ccncc21)C.C1(C(=O)OC(C)(C)C)CCCC1 17618,C1(C(=O)N(CCCN(C)C(C2CC2C(F)F)=O)C)(OC(C)=O)CC1 17619,N1(C(C(c2nc(C(C)(C)C)no2)C)=O)CCCCCC1CO 17620,CC1CN(C(c2coc(C3CCC3)n2)=O)CCN1C(c1cc(Cl)c[nH]1)=O 17621,c1(NC2CN(C(Cc3cc(C)cc(C)c3)=O)CC(F)C2)ncnc2occc12 17622,CC(C)C(C)CC(=O)NC(CN(C)C)C(=O)Nc1cn(C2CC2)cn1 17623,CC(C)(C)C(CNC(C1CC2CCC1CC2)=O)C(=O)N1CCC(CCO)CC1 17624,C1(CNC(c2ccc(C=C)cc2)=O)CN(C(=O)CO)C2(CCC2)C1 17625,C(=O)(C1=C(CC)OCCC1)NC(CC#C)(C)C(=O)N1CCCC(CCO)CC1 17626,C1(C(N2C(CNC(c3c(CC)noc3)=O)CCCC2)=O)Cc2cccc(C)c2O1 17627,N1(C(CCCCCC)=O)CC(C)CN(C(=O)CCC=CC(C)C)CC1C 17628,c1(C(=O)NC(CNC(C2N(C(C)C)CCCC2)=O)C2CC2)ccc(N)c(O)c1 17629,c1(C(N(CC(C)N(C)C(C2CCC(=O)N2)=O)C)=O)coc2c(F)c(Cl)ccc12 17630,CC1CCOC(C(=O)NCCCN(C(=O)Cc2cccs2)C2CC2)C1 17631,c1(C(=O)NC2C(CNC(C3C(CC)CCO3)=O)CCC2)ccc(C2CC2)cc1C 17632,c1(C(=O)NC(C(C)C)CCN(C(=O)CC2CC23CC3)C)ccc(C#N)c(F)c1 17633,c1(CCC)ccc(NCc2ccc(C(C)(F)F)nc2)cc1 17634,C1(C(N2CC3CC2C3NC(C23CCN(CC2)C3)=O)=O)CC12CCCOC2 17635,N1(C(=O)Nc2c(CC)cccc2)CC2CC1CN2C(=O)OC(C)(C)C 17636,C1(C(N2CCC(CCNC(c3ccccc3Cl)=O)C2)=O)CCC2(CC1)CC2(F)F 17637,N1(C(Cc2cc(OC)no2)=O)CC(CNC(=O)C(C)(F)C(C)(C)F)CC(C)(C)C1 17638,N1(C(CCC(N)=O)=O)CC2CC(C1)C2NC(=O)C(Cc1ccccc1)OC1CC1 17639,CC1CCN(C(C2C3CCCC23)=O)CC1OC.C12CC(C1)OCC(=O)O2 17640,N1(C(=O)CCc2ccsc2)CCC(CNC(C2(F)CCOC2)=O)C1 17641,C1(NC(=O)CC2CC(n3cnnc3)C2)(CF)CCN(C(=O)CC2CC2(Cl)Cl)C1 17642,C1(C(=O)NCc2ccc(CNC(=O)COC3CCCC3)cc2)CC2(CCO1)CC2 17643,C1(N(C)C(C2CCC(O)CC2)=O)CCCN(C(=O)CN2CSCC2=O)CC1 17644,c1(CC)nc(C)oc1C(=O)NC(CO)C(=O)NCC1CCCSC1 17645,C(=O)(C1=CC2CCCC12)NCC=CCNC(c1cc(C)c(Cl)s1)=O 17646,N1(C(CC#N)=O)CCC2C(C(=O)NC3CCCCCC3F)C2C1 17647,N1(C(=O)NC2(C)CC2)CCc2c1ccc(F)c2F 17648,C1(CNC(C(c2cn(C)nc2)O)=O)CN(C(=O)Cn2nccn2)CC12CC2 17649,c1(C(NOCC(c2ccccc2)C)=O)cc(O)c(F)cn1 17650,C1(CNC(c2n(CC)ncc2Br)=O)CC2CCC1N(C(=O)C=CCOC)C2 17651,C=CCCCCCCCC(=O)N1CC2(C1)CN(C(c1cn(C3CC3)nc1C)=O)C2 17652,C(CS(=O)(=O)CC(=O)NCc1ccc(C(=O)NCC(CO)C2CC2)nc1)OC 17653,C(=O)(C(O)C(F)(F)F)N1C(C(=O)NCC2(O)CCC2)CCC1C1CC1 17654,C=CC(CC)CC(=O)NC1(c2nnnn2CCCOCC)CCC1(C)C(C)C 17655,C1(C2CCCN(C(=O)C3=C(Cl)CCC3)C2)(NC(C2(C)ON=C(C)C2)=O)CC1 17656,c1(CC)ccc(OCC(=O)NC2CCN(C(C3(C)COC(=O)C3)=O)C2)cc1 17657,c1(C(=O)NCC(CC)NC(C2C(c3ccccc3)C2(C)C)=O)n[nH]cc1[N+](=O)[O-] 17658,C1(CCC(=O)N(C(CCSC)C)C)CCC(NC(c2nccn2C(C)C)=O)C1 17659,c1(C(=O)NCC2N(C(Cc3cnn(C)n3)=O)CC2)cc(=O)oc2ccc(O)cc12 17660,c1(OC)cc(C(=O)NCc2nccnc2Cl)c(NC(C23CC(N)(C2)C3)=O)cn1 17661,C(C)(CO)(C(=O)NCCCN(C(c1cnc(N)cn1)=O)C1CC1)OC 17662,C(=O)(C(C(C)CC)CNC(C)=O)NC1CCN(C(C2(C(=O)OCC)CCC2)=O)C1 17663,N1(Cc2ccc(C(=O)NCc3ccc(CC)cc3)cc2)CCC(C#N)(OC)C1 17664,C(CC(=O)NC1CCCC1NC(c1c(C)nn(C)c1Cl)=O)(C1=CCCC1)OCC 17665,Cc1nc2ccc(C(N3CC(N(C)C(C4CCC4CF)=O)C4(CC4)C3)=O)cc2s1 17666,c1(SC)cc(C(=O)NC2CCC(N(C(=O)C(c3cncn3C)O)C)CC2)n(C)n1 17667,C(=O)(C(C)C(O)C(C)C)N1CCC2C(C(=O)NCC(CSC)OC)C2C1 17668,N1(C(CNS(N)(=O)=O)=O)CC2CCCN(C(c3cc4n(n3)CC(F)C4)=O)C2C1 17669,Cc1ccc(O)c(NC(c2cc(CNC(C3(COC)CCOC3)=O)cs2)=O)c1 17670,C1(C(N)=O)CN(C(c2cnc(Cl)nc2)=O)CC12CN(C(c1cccnn1)=O)C2 17671,N1(C(C=CC)=O)CCC2(CCCC2C(=O)Nc2cccc(Cl)c2F)C1 17672,CC1(C#CC(=O)NCC2CC(CNC(=O)Cn3cnnn3)CO2)COC1 17673,Cc1cc(C(=O)N(CCCN(C)C(C2NC(=O)C3CC23)=O)C)nn1C(C)C 17674,Cn1cnc2nc(N3CCC4CC4C3)[nH]c(=NC3CCCCCCC3)c12 17675,c1(SCC(N2C(CN(C(c3n(C(C)C)ncn3)=O)C)CCC2)=O)cccc[n+]1[O-] 17676,c1(-c2sc(CCOC)c(C)c2)ccnc(OC)c1SC 17677,C1(NC(C(=Cc2cn[nH]c2)C)=O)CCN(C(c2cc(F)c[nH]2)=O)C(C)C1 17678,Cc1cc(C)n(CC(N2CCCC2CN(C(=O)C=CS(C)=O)C)=O)n1 17679,Cc1cc(=O)oc2cc(OC(=O)NOCCC3CC3)c(Cl)cc12 17680,N1(C(c2cnn(CC)c2C)=O)CCCCC(CNC(C2(F)CCOCC2)=O)CC1 17681,c1(C(CC)(C)C)ccccc1C(=O)NCC(C)CNC(c1cn(CC)nc1C)=O 17682,CN=C(NCCCCSC)N1CCN(c2cnccc2C)CC1 17683,n1(CC)cc2ccc(C(N3CC(N(C)C(c4scnc4C)=O)C(O)C3)=O)cc2n1 17684,C=Cc1cc(C(=O)NCC2(O)CCN(C(=O)CC3CCCN(C)C3)C2)cc(F)c1 17685,C12(C(N(C3CCN(C(=O)CN4CCCC4C)CC3)CC)=O)CCC(F)(CC1)C2 17686,CCC(CC(=O)N1CCC(CNC(=O)CNS(=O)(=O)CC)(COC)C1)SC 17687,C(CCN(C)C(C1CCS(=O)(=O)N1)=O)(C(C)(C)C)NC(Cc1c(C)occ1)=O 17688,N1(C(c2c(C)cc(Cl)cc2)=O)CC2CN(C(C34CCCC3C4(F)F)=O)CC2C1 17689,N1(C(C2C(C(=O)OC)C2)=O)Cc2ccccc2CC1C(N1C(C)CCC1C)=O 17690,c1(SCC(=O)NCCOCCCNC(c2n[nH]cc2F)=O)cccc(F)c1 17691,CC12CC(NC(c3cnccc3Cl)=O)(C1)C1(CN(C(=O)CCC3CC3(F)F)C1)O2 17692,c1(-c2cc(C(=O)NCc3cc(Br)ccc3O)c(F)nc2)ccc(F)c2[nH]ncc12 17693,O=C1CC(N=c2nc3scnc3c(NCC3CCCC(O)C3)[nH]2)CN1C1CC1 17694,C(C1c2ccsc2CCN1C(=O)CC(C)CC)NC(CN(CCC#C)C)=O 17695,c1(OC)cncc(C(N2CC(CO)(NC(=O)CNC(C3CCOCC3)=O)C2)=O)n1 17696,N(C1c2ccccc2CC1NC(C1(O)CCSC1)=O)C(C1CCCOC1)=O 17697,N1(C(C(C)C)=O)CCC(C2CC2)(CNC(c2coc(O)n2)=O)C1 17698,c1(OC(C)C)cccnc1C(N1CC2CC2(CNC(C2CC2C)=O)C1)=O 17699,c1(C(N2CCC(O)(CN(C(=O)CNS(N)(=O)=O)C)C2)=O)cc2c(cn1)OCCO2 17700,Cc1ccc(O)c(C(=O)NCc2c(C)noc2C)c1.c12cc(n[nH]1)C(=O)NOC2 17701,C12(C(=O)NCC(CC)NC(=O)COC3CCCCC3)CCC(C1)C(C)(C)O2 17702,N1(S(C)(=O)=O)CCCC(c2n[nH]cc2NC2CC(OC3CNC3)CN2)C1 17703,c1(CC(=O)NCC2OCCN(C(C(=O)N(C)C)=O)C2)c(Cl)ccc(O)c1Cl 17704,C=CC1(C(=O)NCCOCCN(C)C)CCN(C(=O)CC2CCCN2C)C1 17705,c1(C(=O)NC2(COC)CN(C(=O)C(C)(C)F)C2)cc(C)c(OC)c(C)c1 17706,C1(C(=O)NC2(CC(N3CCC(C(=O)NC)C3C)=O)CC2)CCC(=O)N(C)C1 17707,c1(C(=O)NCCCC(C)NC(=O)C(F)C2CC2)ccc(C(F)F)c(F)c1 17708,C1(N(CC=C)C(=O)NCCS(=O)(=O)N(C)C)CCN(C)CC1 17709,N1(C(c2c(C(C)C)c[nH]c2)=O)CCC(F)(F)C(NC(=O)C2CC2)C1 17710,C1(OC)CCC2(C(N3CC(O)CC3CNC(C3(c4cc[nH]n4)CC3)=O)=O)CC12 17711,C(=O)(C(C)(C)CCS(C)(=O)=O)NC(C)CNC(=O)C#CC1CCCCO1 17712,c1(C(=O)NCC(C(C)C)NC(C2CC3CCC2O3)=O)ccc2ncnn2c1 17713,Cc1coc(C)c1C=CC(=O)N(C(C)CCNC(=O)CC(C)(C)CN(C)C)C 17714,C1(CC(=O)NC2CCC2NC(C2CC=CC2)=O)CCCCC1(F)F 17715,C1(NC(CC2(C)CC2)=O)CC2COCC(C1)C2NC(c1cnn(CCO)c1)=O 17716,C(=O)(C1=CC2CCC=CCCC12)N1CCC(NC(CS(=O)(=O)NC)=O)C(C)C1 17717,C(c1ccccc1F)=CCC(=O)NCC(CC)(C)NC(c1cnc(O)n1C)=O 17718,CC(C(=O)N1CC(O)CC1CC(N1CC(C(=O)N(C)C)C1)=O)S(C)(=O)=O 17719,C1(NC(CC(=O)NCC#C)=O)CC2CCC(C1)N2C(C12CCC(F)(CC1)CC2)=O 17720,c1(C(C(N2CC3=C(CN(C(C)=O)C3)C2)=O)=O)c(C)[nH]c2ccccc12 17721,C(c1ccc(C(F)(F)F)cc1)=CC(=O)NC1(C)CCN(C(c2ccsn2)=O)C1 17722,c1(C2CC(C(N(CC(C)N(C)C(c3c[nH]c(=O)cn3)=O)C)=O)C2)ccc(Cl)cc1 17723,c1(C(=O)NC2CC(OCC(=O)N(CCCOCC)C)C2)ccc(C)cc1CC 17724,C12(NC(Cc3cn(CC)nc3)=O)CCC1CN(C(=O)C=CC1CCOCC1)C2 17725,CC1=C(C(=O)NC(C2CCN(C(=O)CCCc3ccncc3)C2)C)CCO1 17726,C(=O)(C(F)(F)CCn1cccn1)N(CCCn1cc(C(CC)O)nn1)C1CC1 17727,C(c1ccc(O)cc1)=C(C)C(=O)NOCc1cc(-c2cccnc2O)ccc1OC 17728,CC1(C)CN(C(=O)CC2OCCCO2)CCC1C(=O)NCCC(O)C(F)(F)F 17729,C1(CC)(NC(=O)Cc2cnoc2)CCN(C(=O)C(O)CC2CCOCC2)CC1 17730,C1(O)(C(CNC(c2c(C)scn2)=O)C)CCN(C(c2cnn(C)c2Cl)=O)C1 17731,Cc1noc(C)c1C(C)CC(N1CC(C(F)(F)F)C(C(F)(F)F)C1)=O 17732,C(=O)(CCCC(C)(C)C#N)N1CC(NC(C2(CC)CCCC2)=O)C(C)C1 17733,c1(C(C)OC)nc(C)c(C(N2CCCC(CNC(C3CN(C(C)C)C3)=O)C2)=O)s1 17734,c1(C(=O)NCC2CN(C(CCOCCOC)=O)C2)ccc(N)c(C)c1Cl 17735,c1(CC2(C#CC(=O)NCC3C(CC)CCCC3)CC2)c(OC)nc(C)nc1Cl 17736,c1(OC)c[nH]nc1C(=O)N(C(CNC(=O)CN1CCCC1C)C1CC1)C 17737,Cc1cn(C)cc1C(=O)NC1C=CC(C(=O)NCCC(=O)NCCN(C)C)C1 17738,C1(C(=O)NCCOC2CCC2)CN(C(C2CC23CC3)=O)CC1F 17739,C(=O)(C(N)CCC(=O)N1CCCC(C(N2CCC(C(N)=O)CC2)=O)CC1)OC 17740,N1(C(COCC=C)=O)CC2(CCC2CNC(=O)C(=O)NOC)C1 17741,c1(C(N(C(c2ccccn2)C)C)=O)c[nH]n(C)c1=O 17742,CC(C(C)(C)NC1COCC1C(=O)OC(C)(C)C)NC(=O)C(N1CCC(C)C1)=O 17743,Cc1nc(C(N2CCS(=O)(=O)CC2C(=O)OC(C)(C)C)=O)c(=O)[nH]c1C 17744,Cc1nc(C2CN(C(=O)C(C3CCCO3)NC(=O)CCNC(N)=O)C2)n[nH]1 17745,N1(C(c2ccc(C(C)C)cn2)=O)CCC2(NC(c3cn(C)ccc3=O)=O)CC2C1 17746,c1(CCC(=O)OCC)cc(=NC(C)CC(C)NC(=O)C(C)SC)[nH]c(C)n1 17747,C1(C)(C(N2CC(O)(CN(C(=O)Cc3n[nH]c(=N)s3)C)C2)=O)Cc2ccccc2C1 17748,N(C1COc2ccccc21)C(C1N(Cc2cc(OCC)c(O)c(Br)c2)CCC1)=O 17749,N1(C(CCC2(NC(C3C(C(=O)OC)C3)=O)CCCC2)=O)CC2C(=O)NC(=O)C2C1 17750,C1(CC(=O)NCc2ccccc2F)C2CN(C(=O)CC3CCOC3)CC12 17751,C1(C(=O)NCc2cc(C)ns2)CN(C(=O)CCc2cc(C)[nH]n2)CCO1 17752,C(=O)(C(C)(C)C(=O)N(C)CC1CCCN1C(=O)CCc1csc(C)n1)NC 17753,C(=O)(C(F)(CNC(=O)C1=CCN(C)C1)C(C)C)N(C)Cc1cccc(C)n1 17754,N1(C(C2CC(=O)NCC2)=O)CC(NC(=O)CCc2cnc[nH]2)C(F)(F)C1 17755,CCCC(C)(C)C(=O)NC1CCCC1CC(=O)NCC(=O)N1CCCO1 17756,c1(C(=O)NCC(CNC(=O)COCC2CCC2)CO)cc2c(s1)COCC2 17757,C(=O)(C1=C(Cl)CCCC1)NC12C(CN(C(C(C(C)C)n3cnnn3)=O)C1)C2 17758,CC(CC1(C)OCCO1)CN=c1[nH]c2c(c(=NCc3nccs3)[nH]1)SCC2 17759,C12(C(N(C3CCN(C(=O)C(O)c4ccsc4)CC3)C)=O)CCCC1CC(=O)CC2 17760,C1(CNC(C2(C(=O)NC)CCC2)=O)C2CCC(C2)N1C(c1ccc(C(N)=O)[nH]1)=O 17761,N1(C(C2C(C)C2(F)F)=O)CCN(C(c2cscc2C(F)F)=O)CC(C)(C)C1 17762,C1(CN(CC(C)(O)CCC2CCCCC2)C(=O)OC(C)(C)C)CCCC2(CC2)C1 17763,CC1CC(C)C1C(=O)N(C)CCN(C)C(C1(C(N)=O)CC1)=O 17764,Cc1ccc(C(=O)NCCC2CCN(C(C3CCOC3=O)=O)C2)c2ncccc12 17765,N1(C(C2(COC)COC2)=O)CCCC(O)(CNC(c2cn(C3CCC3)nn2)=O)C1 17766,N1(C(C)=O)CCc2sc(S(=O)(=O)NCc3cc(C(C)(C)C)no3)cc2C1 17767,CC1CN(C(C2CCCC(CF)C2)=O)C(C)CN1C(=O)CC1CSCCO1 17768,C1(C(=O)NCCCCCC=C)CCN(C(=O)C(C)(C)C(F)F)CC1C 17769,C(CCCC(C)(F)F)NC(CNC(C(c1ccnn1C)C)=O)=O 17770,CCCCC(C)C(=O)N1CC(CNC(=O)CCOCC)C(O)C1 17771,Cc1c[nH]c(C#N)nc1=NCCNC(C1COc2ccc(F)cc2C1)=O 17772,C1(NC(C(C)NC(N)=O)=O)CCN(C(=O)CCCc2csc(=N)[nH]2)C12CC2 17773,c1(C(=O)NC(c2cn(C(C)C)nn2)CCC)ccc(Cl)cc1-n1cncn1 17774,N#CC1CN(C(c2ccc(S)cc2)=O)CC1NC(c1cccnc1)=O 17775,c1(C(N(CCCCCC)C(=O)CN(C)Cc2ccco2)=O)ccc(OC)cc1C 17776,CC(C)C(O)CC(=O)N(C1CCN(C(C23CSCC2C3)=O)CC1)C 17777,C1(CC(=O)NCC(CC)C)CN(C(c2c(C#N)cnn2C)=O)CC12CC2 17778,c1(C(c2n(CC)nnn2)NC(C2CCC2)C2CC2)ccc(OC)cc1[N+](=O)[O-] 17779,C1(NC(C=C(C)C(C)C)=O)CCCCC1CNC(c1ccno1)=O 17780,C1(C(=O)NC(CNC(c2ccc(C(F)(F)F)s2)=O)C2CC2)CCCCS1 17781,n1(CC)nnc2c1CCC(C(=O)NCC1CCN(C(C3COC(=O)N3)=O)CC1)C2 17782,c1(C(=O)NC2(CCNC(C3C(C(=O)OC)C3)=O)CC2)cccc2c1NC(=O)CO2 17783,C(=O)(C(CC=C)CC=C)NCC1C2CN(C(COc3ccc(C#C)cc3)=O)CC21 17784,c1(C(N2C(C(=O)NCC(C)CC3CC3)C=CC2)=O)cc(F)ccc1O 17785,C1(NC(c2ccc3occc3c2)=O)CN(C(C2CC2CF)=O)CC2(CCC2)C1 17786,n1(CC)cc(-c2ccc(CC(=O)N(CC)Cc3ccncc3)nc2C)ccc1=O 17787,c1(C(N2CCC(NC(c3cncc(OC)c3)=O)C(O)C2)=O)ccc(P(C)(C)=O)o1 17788,c1(C(=O)NCCOCCC(=O)NCC2(SCC)CC2)ccc(C)cc1C 17789,C(=O)(CCS(=O)(=O)N(C1CCC(NC(=O)CCc2ncc(C)[nH]2)C1)C)OC 17790,O(NC(=O)C(C)(C)C1CCCN1C(=O)CCNC(=O)NC)CC#C 17791,C1(NC(C=Cc2nc(C)sc2)=O)CC(CNC(=O)CC2(O)CCC2)C12CCC2 17792,c1(C(=O)Nc2c(C(C)(C)C)ncs2)cnc(C2CCNCC2)nc1 17793,N1(C(c2cn(CCC)nn2)C(=O)NC2CCCC2)C2CCC1CN(C)CC2 17794,C1(CC(=O)Nc2ccc(Br)nc2)COCCN1Cc1ccc(-c2ccccc2)s1 17795,CCCCC(C)(F)C(=O)N1CC(NC(C23CC(C)(C2)OC3(C)C)=O)C(O)C1 17796,C(=O)(C(CN(C)C)CC)NC(c1ccccc1N(C)C)CNC(C1C(=C)C1)=O 17797,c1(C2(N(C(=O)Cn3cc(C(F)(F)F)cn3)C(C)C)CC2)ccnc2ccccc12 17798,C12(C(=O)NC)CCCCC1CN(C(c1c(C(=O)OC)cccc1[N+](=O)[O-])=O)C2 17799,N1(C(C2CCC(CC)O2)=O)CC2(C1)CN(C)CC2c1cc[nH]c(=NCCC)n1 17800,N1(C(CSCC)=O)Cc2ccccc2CC1CNC(c1cc(Cl)ccc1OC)=O 17801,NC(=O)CCCC(=O)N1CCC(C2OCCC2Cc2ccccc2)CC1 17802,CC1CCN(C(=O)Cc2cncc(C(F)(F)F)c2)CC1c1ccc(F)cc1 17803,CCC(C)CCCCC(=O)NC(C)CNC(c1ccc(S(C)=O)cc1)=O 17804,CN1CCN(c2ccc(C(N3CC(NS(=O)(=O)CC4CC4)C(O)C3)=O)cc2)CC1 17805,c1(C(N2CCC(C(=O)NCC3CC(C4CC4)=NO3)CC2)=O)[nH]nc([N+](=O)[O-])c1Br 17806,c1(C(N2C(CNC(=O)CCC3NC(=O)NC3=O)CCC2)=O)ccc(CO)cc1F 17807,N1(C(c2c(C)c[nH]n2)=O)CCCC(NC(c2ccsc2Cl)=O)C1C 17808,c1(NCC(CC)CCO)cc(S(=O)(=O)NCC2CCC3(CC3)C2)ccc1C#N 17809,CN1CCC(C(=O)NC2CCC3(CC3)C2)(NC(C2C=CCCC2)=O)C1 17810,C1(C(=O)NCCOCCCC#C)CCN(C(C2CC(C)CCO2)=O)C1(C)C 17811,C1(C(=O)NC(C(C)C)CCNC(=O)C=Cc2cnn(C)c2)CCC2(C1)CC2(F)F 17812,C1(C2CC2)(CNC(c2c(CCC)n[nH]c2)=O)CCN(C(=O)CC(C)(F)F)C1 17813,C(=O)(CCCC(c1nnnn1Cc1ccccc1OC)Nc1ccc(F)cc1F)OC 17814,C(=O)(CCCC(F)(F)F)NC(CN(C)C)C(N1C2CCC1CC2)=O 17815,C1(F)(CNC(c2cccc(CCC)c2)=O)CCN(C(=O)C(F)=CC2CC2)CC1 17816,c1(Cn2cc(-c3c(C)ocn3)nn2)cccc(C(=O)NCC2CSCCS2)c1 17817,c1(NC(CN2CCCC(C)C2)=O)ccc2nn[nH]c2c1 17818,C(=O)(C(CC)CCOC)N(CCC(=O)NC(c1ncc[nH]1)C)CC#C 17819,C1(F)(CNC(=O)CSC(F)(F)F)CC2CCC(C1)N2C(=O)CC1CS(=O)(=O)C1 17820,Cn1cnc(NC2CC(NC(C3CC34CC(C)(C)C4)=O)C2)cc1=O 17821,c1(C(=O)NC2C(CNC(C(COC)(F)F)=O)CCCC2)cnc2c(c1)CCC2 17822,c1(N(C)C)cccnc1C(=O)NCCC1(CNC(=O)C(C)(C)c2cncs2)CC1 17823,C1(C)(CCCC(=O)NCc2ccc(C(=O)NCc3cc(C)sc3)o2)NC(=O)NC1=O 17824,S(=O)(=O)(c1cnc(C(C)(C)C)[nH]1)N(C1C(CCC)C1)C 17825,NS(=O)(=O)c1cc(C(=O)NC(CNC(c2cncc(Cl)c2)=O)C2CC2)ccc1Cl 17826,c1(CC(N2CCC(C(C)C(=O)NC3CC(F)C3)CC2)=O)ccc2c(c1)CCCO2 17827,c1(C(N2CCN(C(c3ccn(COC)n3)=O)C(C)C2)=O)c(C)cc(O)nc1C 17828,N1(C(CCC(C)N(C)C)=O)CCC=C(C(=O)N2CCC(C)(C#N)CC2)C1 17829,Cc1ccc(CC(=O)NCC2CC(CNC(c3ccc(C(F)(F)F)s3)=O)CO2)o1 17830,c1(OC(CC)CC)ccc(C(=O)NCC2CC2CNC(c2cn(C)cn2)=O)cc1 17831,C1(N(C)C)(C(=O)NCC(CNC(=O)Cc2nc(C3CC3)cs2)CO)CCCSC1 17832,c1(C(N2CC(COC)N(C(C3CCC(C)(C)O3)=O)CC2)=O)ccc2cc[nH]c2n1 17833,C1(NC(CC2(C(=O)OC)CC2)=O)CCCCN(C(C2CC(F)C2)=O)C1 17834,N1(C(CCCOC(C(C)C)=O)=O)CCCC(C(=O)Nc2cccc(O)c2)C1 17835,c1(C(N(CCCCNC(c2c(C)nccc2Cl)=O)C)=O)oc2ccccc2c1C 17836,C1(C(=O)NCC2CC2NC(C2CS(=O)(=O)C2)=O)CCCC1C(F)(F)F 17837,C1(C)(C(=O)NC2(C)CN(C(=O)CC(C)(O)c3ccccc3)C2)CCCCNC1=O 17838,CC(C#N)C(=O)N(CC(O)CN(C(=O)CN(CCc1ccccc1)C(C)=O)C)C 17839,C1(CCOC)(C(=O)N(CCCO)C)CCN(C(=O)CN(C)C2CC2)C1 17840,C#CCCCC(C)C(=O)NCc1ccc(C(N2CCCC(C)(C)C2C)=O)cn1 17841,N1(C(C(CC)(C)C)=O)CCN(C(C2CCCC23CCC3)=O)C(C)C1 17842,c1(C(=O)NC2(C)CC(NC(C3N(C(C)=O)CC(O)C3)=O)C2)cc(O)cc(C#N)c1 17843,Cn1cnc(C=CC(=O)NCC(=O)NC2CC(O)C(F)C2)c1 17844,n1(CC)cc2ccc(C(N3CC4CCOC4(CNC(=O)CSC)C3)=O)cc2n1 17845,c1(C(=O)NC2CCCC(NC(C(C)(C)C3CCOCC3)=O)C2)c[nH]cc(F)c1=O 17846,c1(-n2c(CCS(CC)=O)nc(CCC(C)C)n2)nc2ccccc2n1C 17847,Clc1ccc(C(c2nnnn2CCCl)NCc2ncoc2CN2CCOCC2)cc1Cl 17848,c1(CNC(C2CC(C)(C)C2)=O)cccc(NC(=O)CCc2ccsc2Cl)c1 17849,C1(C)(CC(=O)N(CC(n2ccnc2)C)C)CCN1C(=O)COC1CCCCC1 17850,C1(NC(C(C)NC(=O)NC)=O)CN(C(c2cc(C)co2)=O)Cc2nccn2C1 17851,C1(c2cn(CCOCC)nn2)CN(C(=O)Cc2csc(C)c2C)CC1C 17852,c1(-n2cc(C3CN(C(C4C(CC)CCC4)=O)C3)nn2)cc(F)ccc1C 17853,N1(C(c2ccc(OC)cc2)=O)CCN(C(c2cc(OC)no2)=O)C(CF)C1 17854,c1(OC)cc(C(N2CCC(NC(=O)C=CC(C)(C)C)C(CO)C2)=O)ccc1C 17855,c1(C(N2C(C)CN(C(=O)C(N3CCOCC3)C)CC2)=O)cn2cnnc2cn1 17856,C1(CCNC(c2[nH]cc(C)c2C)=O)CCN(C(=O)C(C)n2ccnc2)CC1(F)F 17857,N1(C(C(C)C(F)F)=O)CCC(F)(C(N2CCC(C(C)(C)C)CC2)=O)CC1 17858,C(c1cccs1)=CC(=O)N(CC(CC)NC(=O)CC1CCOC1)C 17859,c1(C(=O)NCC2N(C(C(C=C)OC)=O)CC(F)C2)cc(C)c(C#N)c(C)c1 17860,C=CCC(C(=O)NC(C=C)CO)NC(=O)C=CC1CCCN1C 17861,C1(CNC(CSCC=C)=O)CN(C(C2COCOC2)=O)CCC1C 17862,CN1CC(NC(=O)CC2CC(F)CN2C(=O)CC2CCCC2O)C2(CC2)C1=O 17863,C=C(C)C(C)(C)C(=O)NC(C1CCCN1C(c1ccoc1Cl)=O)C 17864,CC1CC(NC(=O)Nc2nccc(-n3cccn3)n2)CCN1C 17865,c1(C(C)=O)c(C)[nH]c(C(=O)NCCC2(O)CN(C(=O)C(C)N=[N+]=[N-])C2)c1C 17866,N1(C(COCCCCC)=O)CCC(CC)C1CNC(=O)Cn1cnc(C#N)n1 17867,C1(C(=O)NCC2CC(CNC(C(Cc3ncn(C)c3)O)=O)C2)Cc2nccn2C1 17868,c1(OC)ccc(C(=O)NC2CCC(NC(=O)C(C)(CO)CO)C2)cc1O 17869,C1(COC)CN(C(=O)C(C)C#N)CCN1C(=O)CCc1cnc(O)[nH]1 17870,c1(CNC(CSCC(=O)N(c2ccccn2)C)=O)ccc(Cl)cc1 17871,C(=O)(C1CCc2c[nH]nc21)NC1CCC(CC(=O)N(c2cccc(O)c2)C)CC1 17872,C1(C(=O)NCC2CCN2C(=O)C(F)(F)CC2CC2)CCC([N+](=O)[O-])CC1 17873,CCC(CCOC)NC(C1CC(NC(=O)C(F)OC(F)(F)F)C1)=O 17874,Cc1nc(Br)oc1C(=O)NC(C)CN(C)C(c1cc(C(C)(C)C)n[nH]1)=O 17875,c1(CC=CC(=O)N(C(CNC(C=CC(CC)=CC)=O)C)C)ccccn1 17876,C1(C(N(CC(CNC(c2c(OC)c(Cl)ncc2)=O)C)C)=O)OCCOC12CCC2 17877,N1(C(c2n(C(C)C)ccn2)=O)C2CCCC1CN(C(C1CCCSS1)=O)C2 17878,N1(C(CC(CC)OC)=O)CCC(C2(O)CN(C(C3(CO)CCC3)=O)C2)CC1 17879,N1(C(c2ccc(C)nc2C)=O)CCC2C(CCN2Cc2cc(Br)cc(Cl)c2O)C1 17880,CCC(C)CC(=O)C(=O)N1CCOC(C(=O)NCC2(C)C=CCCC2)C1 17881,N1(C(C(=O)N(C)C)=O)CCCC2(C1)CN(C(c1c(F)cccc1F)=O)CCO2 17882,Cc1csc(C(=O)NCC2(CNC(=O)C(F)F)CC2)c1Cl 17883,c1(C(=O)NC(CC=C)CNC(=O)Cc2csc(=N)[nH]2)nn(C)c(Cl)c1Cl 17884,C1(C(N(CCN(CC=C)C)CC)=O)C=CCN(C(=O)C(C)(O)C2CCC2)C1 17885,C1(C)(CC)CCN(C(C2(N(C(=O)CCc3ccoc3)C)CC2)=O)C1 17886,C1(NC(c2ccc(Cl)nc2Cl)=O)CCN(c2ncncc2I)CC1F 17887,O=C1NC2CCC1CN(S(=O)(=O)c1ccc(N3CCCC(C(F)F)C3)nc1)C2 17888,S(=O)(=O)(c1cc(F)ccc1OCC1CC1)N1CCC(C)(CC(F)(F)F)C1.OC 17889,N1(C(c2c(C(C)C)nns2)=O)CCC(CNC(C2(C#N)CC3CC3C2)=O)C(C)C1 17890,C1(CNC(CN(C)C)=O)(CNC(=O)C2CC2)CN(C(=O)COc2cccnc2)C1 17891,c1(C(N2CCCC(c3ncc[nH]3)C2)=O)cccc(-n2cnnn2)c1 17892,c1(C(N2CCC(OC)C2)=O)cnc2c(c1)CCN(Cc1cc(Cl)c(O)c(Br)c1)C2 17893,c1(C(=O)NC2CN(C(CC(C)SC)=O)CC23CC3)ccn2ccnc2n1 17894,c1(OC)ccc2c(c1)CCC2C(=O)N1CC2(CCCC2(F)F)C1 17895,C#Cc1ccc(F)cc1C(=O)NCCC(C)(C)NC(c1cn(C(F)F)c(C)n1)=O 17896,N1(C(CC)=O)CCCC(C(=O)NC(CNC(c2ocnc2C(F)F)=O)C2CC2)C1 17897,N(C1CC2(CC2)Oc2c(F)cccc21)C(C1(F)CC=CCC1)=O 17898,C12(CNC(CCC=C)=O)CC1CN(C(c1cc(C(=O)OC)sn1)=O)C2 17899,c1(SCC)cccc(CC(=O)NCC(CC)NC(c2ccc(C(F)F)nc2)=O)c1 17900,Cc1cc(C)c(C(N2CCC(N(C)C(c3cn(C(C)(C)C)nc3C)=O)C2)=O)cn1 17901,CCCCCC(=O)N(CCCNC(c1ccc(-c2nc(C)no2)cc1)=O)C1CC1 17902,N1(c2nnc(CCC)o2)CCCC(C(N2CCC(C(=O)O)CC2)=O)CC1 17903,C1(NC(Cc2ccc(C(C)=O)s2)=O)CN(C(c2ccccc2)=O)CC1C 17904,CC#CCCCC(=O)NCC1(F)CC(NC(=O)Cc2noc(C)c2C#N)C1 17905,N1(C(C2C(C(C)C)C2)=O)CCC(C)(CCNC(c2cc(Cl)n(C)n2)=O)C1 17906,C1(NC(N2CCC(C(=O)OC)(CF)C2)=O)CCC(C)(C)CC1Cc1ccc[nH]1 17907,C1(COC)CN(C(=O)CC2CCCCC2(C)C)CCN1C(=O)CC(=O)OC(C)(C)C 17908,N1(C(CC(C=C)C)=O)CC2(C1)OC1(CO)CC2(NC(=O)CC2CC(OC)C2)C1 17909,C1(CC)CCCN(C(=O)C(n2ccnc2C)C)C1C(=O)NC1COCC(C)(C)C1 17910,Cc1cc(C(N2CCC3(C2)CN(C(=O)C(C)C(F)(F)F)C3)=O)c(Br)c(C)c1 17911,c1(NC(C2N(C(CCc3ccc(C)cn3)=O)CC2)=O)ncc([N+](=O)[O-])cc1I 17912,c1(C(=O)NC(C(C)NC(C2CCOCC2(C)C)=O)CO)cc2cc(Cl)cnc2[nH]1 17913,c1(Cn2cc(COC)nn2)cc2cc(C)cc(C)c2[nH]1 17914,CC1CN(C)C(C)CN1C(C1CC2CCC1N2C(=O)NC1(c2cccs2)CC1)=O 17915,c1(C(=O)NCC(C)(CO)NC(C2N(C)CC(O)C2)=O)cc2ccncc2s1 17916,Cc1ccc(C(=O)NCCCC(O)C(=O)N(c2csnc2C)C)c(O)c1 17917,c1(C(=O)NC2CCC(C)(CNC(C3C(C)=C3)=O)C2)cc(C)nc2onc(C)c12 17918,c1(C(=O)NC2C(C(N3CC(SC)C3)=O)COCC2)ncnc(O)c1F 17919,C1(C(=O)NCC2CC(NC(C(Cn3ccc(C)n3)C)=O)C2)CCC(=O)NC1 17920,C1(CC(=O)NCC2C(NC(COCC(C)C)=O)C2)CC(OC(C)(C)C)C1 17921,c1(OC(C)C)ccc(CC(=O)NCC2(CNC(=O)CSC3CC3)CC2(F)F)cc1 17922,c1(C(=O)NC(C(C)NC(C(CC#C)O)=O)(C)C)[nH]cc2c1CCCC2 17923,c1(C(N2C(CN(CCCC3CCOC3)C)CCCC2)=O)cc2sccc2[nH]1 17924,N1(C(Cc2nc(C)sc2)=O)CCC(O)(C(C)CNC(c2ccnc(CO)n2)=O)C1 17925,C1(C)(C(N(CC(C)(C)NC(C(c2ccc(Cl)s2)C)=O)C)=O)CC2CC2C1 17926,CCCC(C(=O)OCC)N1CC2C(C1)N2C(=O)CCCO 17927,c1(CC(=O)NC2C(SC)CN(C(c3cnc(O)o3)=O)C2)ccc2c(c1)NC(=O)C2 17928,N1(C(CCSC)=O)CCN(C(C2(CO)CCC2)=O)CC1c1ccccc1Cl 17929,c1(OC)nc(Cl)ccc1C(=O)NC(C)CC1CN(C(=O)C(c2ccc(Cl)s2)C)C1 17930,c1(N2CCC(CC)CC2)[nH]c(=NC(CCO)CC(C)C)nc2c1ncn2C(C)C 17931,C1(O)(C(C(=O)NCC=C)NC(=O)C=CCC2(SC)CCC2)CCCCC1 17932,C#CCC(CC(F)F)C(=O)N1CCCC(O)(C(C)NC(=O)CC(=O)NCC)C1 17933,c1(N(C(CNC(C(C(C)C)OC)=O)C)C)cc2nnc(-c3ccccc3)n2cn1 17934,C(=O)(C1Cc2c(Cl)cccc21)NCCC1(C)CCN(C(CCCOCC=C)=O)C1 17935,c1(NC(C=CC2N(C(CN3CCC(OC)C3)=O)CCC2)=O)ccc(Cl)nc1C 17936,N1(C(C(C=C)(C)C)=O)CC(NC(c2cc(C(C)C)on2)=O)CC2(CCC2)C1 17937,N1(C(c2n(C(C)C)ncc2)=O)CCOC(C)(CNC(c2nn(C)nc2Br)=O)C1 17938,C1(CNC(=O)NC(C)COC(F)(F)F)Cc2ccc(F)cc2C1 17939,C12(C(N3CCC4(NC(=O)C=Cc5ccco5)C(C3)C4)=O)CCC(F)(CC1)CC2 17940,Cc1ccc(-n2cc(C(=O)NC(Cc3cncn3C)C(=O)O)cn2)cc1 17941,N1(CCC(=O)NCCOCCCNC(C2(F)CC2)=O)C(=O)C2CCCCC2C1=O 17942,C1(C(N2CCC(C)C2)=O)C2C3CCC(C3)C12.C1(=O)CCC2(CCC2)N1 17943,Cc1ccc(Cl)c(C(=O)NCC2CCCCN2C(=O)Cc2cc(C)ccc2C)c1 17944,c1(C(C)C)ccc(C(=O)NCC2C3CCC(C3)N2C(C2(C)CCOC2)=O)c(F)c1 17945,c1(CC(N2CCC(NC(c3c(CC)c[nH]c3)=O)(CF)C2)=O)cc2ccccc2o1 17946,c1(C(=O)NCC2N(C(c3c(CC)cno3)=O)CC(OC)C2)c[nH]c(=NCC)s1 17947,N1(C(C(CC)SC)=O)C(C(N2CCC(C(=O)OC)C2(C)C)=O)CCC12CC2 17948,Cc1ccncc1-c1cn(C(C)C(N2CCCC(C(=O)NC3CC3)C2)=O)nn1 17949,Cn1c(CN2CCCC3C(=O)NCC23)c(Cl)c2ccccc12 17950,N1(C(CC(=C)C)=O)CC2CC(NC(c3cc(OC)cs3)=O)C(C2)C1 17951,N1(C(COCCN(C)C)=O)CC(C)(NC(=O)Cc2csc(S)n2)C1 17952,c1(C(=O)NCCCCCNC(c2cncc(N)n2)=O)ccc(S(N)(=O)=O)cc1Cl 17953,c1(CC)cc(C(=O)NCCNC(=O)COCc2cccc(C)c2)nn1C 17954,C1(C(=O)NC(c2cnc(C)s2)C)CCC(C)(C)N(C(=O)CC2=CCCCC2)C1 17955,c1(C(=O)NCC2C(NC(C=C(C)C(C)C)=O)CC2)ncnn1C1CCOCC1 17956,N1(C(C=Cc2nc(C)sc2)=O)CCCCC1C1CCCN1C(=O)C(F)C1CCC1 17957,n1(C(C)C)cc(C(=O)NCCC(C)N(C)C(c2cc(F)n[nH]2)=O)c(Br)n1 17958,C(=O)(C(C)(C)C(=O)c1ccccc1)N(CCC=C)C(=O)CN(CCOC)CC 17959,c1(C(N(CC(C)NC(c2n(CC)ccc2)=O)C)=O)cc(Cl)ccc1F 17960,C1(O)(CN(C(C2C(COC)CC2)=O)C)CCN(C(=O)C(C)N2CC(C)C2)CC1 17961,c1(C(=O)NCCCNC(c2cn(C3CCC3O)nn2)=O)cc2ccsc2s1 17962,C1(C#N)(C(=O)OC)CC2CCC1CC2NC1CCCC1Cc1ccccc1 17963,C1(NC(CN(C(COC)=O)C)=O)CC2CC1CN(C(=O)Cn1ccnc1C)C2 17964,CC(C(=O)NCC1CCN(C(=O)Cc2cncs2)CC1CO)C(F)(F)C(F)F 17965,c1(C(N(C2CCCN(C(=O)C(O)C3CCCC3)C2)CC)=O)cc2cnccc2o1 17966,C1(NC(C(C)SC)=O)CC2(CCCN(C(=O)C(F)C(C)(F)F)C2)C1 17967,C=C1CCN(C(c2sc(C)cc2C)=O)C(C(=O)NCCOCCOC)C1 17968,c1(C(=O)NCCC2(C(=O)NCCCCN=[N+]=[N-])CCCC2)ccc(O)cc1F 17969,CNS(=O)(=O)NCC(=O)NCCOCCNC(=O)Cc1conc1C 17970,C1(C(N2CCCC2)CC)CCCN(c2cccc(C(N)=O)n2)C1 17971,N1(C(CCCNC(=O)OC)=O)CC(O)CC1(C)C(N1CCC1CF)=O 17972,Cn1cccc(-c2cccc(C3CC3C(=O)Nc3ncc(Br)nc3Cl)c2)c1=O 17973,C1(O)(C(C)NC(C2CN(C)C(=O)N2)=O)CCN(C(c2scnc2C(F)F)=O)CC1 17974,n1(CCNC(c2cn(C)nc2I)c2nnnn2C2CC2)cc(Br)ccc1=O.C1(C)CC1 17975,C(c1ccc(F)cc1)=C(C)C(N1CCC(C)(NC(=O)CN2CCCCS2(=O)=O)C1)=O 17976,c1(-c2cn(CC(CN)OC)nn2)ccc(C(F)(F)F)cc1Cl 17977,C(=O)(C(C)CC(F)F)NC(CN(C(c1ccc(C(C)C)cn1)=O)CC)C 17978,N(C(=NCCCN1CC(C)OC(C)C1)N1CCN(C2CC2)C(=O)C1)CC(=C)C 17979,c1(C(N)=O)ccc(C(=O)NCCc2cn(CCNC(N)=O)nn2)cc1 17980,C=CC(C)(C)CC(=O)N1CCC(CO)(NC(=O)C(CC2CCCCC2)CCC)C1 17981,Cc1ccn(C)c1C(N1CC(O)(CN(C(=O)CCc2ccnc(Cl)c2)C)C1)=O 17982,C(=O)(C1=CCC2CCC1N2C(=O)C(Cl)Cl)NC(c1ccco1)C 17983,c1(CC)ccc(N)c(C(=O)NCC2(NC(=O)C=Cc3ncc[nH]3)CCOCC2)c1 17984,c1(OC)cc(CC(=O)NCC2CCCN2C(=O)Cc2cc(C)[nH]n2)c(F)cc1O 17985,C1(NC(CCCC#C)=O)CCCC12CN(C(c1cccnc1OCCOC)=O)C2 17986,C1(NC(CCOCC#C)=O)CC2(C1)CC2NC(c1cnn(CCN(C)C)c1)=O 17987,C1(CNC2CC(CNC3(CC(=O)OC)CCC3)C2)CCCC1C 17988,c1(C(=O)NCC2C(NC(CC(C=C)C)=O)CCCC2)ccc(C(F)(F)F)c(N)c1 17989,C1(NC(CCC2(C)CC2(F)F)=O)CN(C(=O)Cc2cccc(O)c2)CC1F 17990,c1(-c2scc(C)n2)ccc(C(=O)N(C2CN(C(C3(C)CCCN3C)=O)C2)C)cc1 17991,c1(C(N2CCC(NC(CCC(CC)C)=O)(COC)C2)=O)cnc2ccccn12 17992,N1(CC(=O)N(c2nc3ccccc3o2)CC)CCC(C2CC(F)(F)C2)C1 17993,c1(C(=O)NCC(c2ccc(C)cc2)NC(C2(C3CC3)CC2)=O)cnc2n1CCS2 17994,CC1CN(C(c2cn(CCNC(=O)C(C)(Cl)Cl)cn2)=O)CC1(C)CO 17995,C(=O)(CCCC(F)(F)CO)NC1C(SC)CN(C(c2c[nH]nc2[N+](=O)[O-])=O)C1 17996,N1(C(=O)Cc2ccc(Br)cn2)CCC(F)C(NCc2cc(O)cc(F)c2)C1 17997,N1(C(C2C(C)CCO2)=O)CCC(F)(C(N2CC(C3CCCO3)C2)=O)C1 17998,N1(C(C(c2cn(CC)nc2)(F)F)=O)CCC(O)C(NC(c2nnn(C)c2C)=O)C1 17999,CC1CC(C(=O)NOCC(=O)NCCN2CC=CC2)CC(=O)N1 18000,N1(C(Cc2cc(C(=O)OC)sc2)=O)CC(NC(c2ccc(C(N)=O)[nH]2)=O)C(C)C1 18001,C1(C(C)NC(=O)Cc2cnc[nH]2)CCCCN1C(c1ccc(C2CCC2)cc1)=O 18002,c1(Cn2cc(C3(O)CSC3)nn2)ccccc1C1(NC(C2CC3CC3C2)=O)CC1 18003,CC1(C)C(CC(=O)NCc2nc(C3CC3)cs2)CCN1C(=O)CC1(C#N)CC1 18004,C1(NC(CCCN(C(C)C)C)=O)CCCN(C(=O)CN2CC3CC3C2)C1C 18005,C1(C(N2CC(C#N)C2)=O)CC(OC)CCN1C(C1CC2CCC(C1)C2)=O 18006,c1(CNC(C(C)(C)NCC2(F)CCN(C(C)C)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 18007,N1(C(C2(F)CN(C(CS(CC)=O)=O)C2)=O)CC(C)OC(C)(C)C1C 18008,c1(-c2cncc(OC)c2)ccc(CN2CCCC2(C)CO)c(C)c1 18009,C(=O)(C1(C)CCn2c(C)nnc21)N1CC(NC(c2ncc(C)cn2)=O)C(O)CC1 18010,c1(C(=O)NC2CCCC3CN(C(CCSC)=O)CC32)cccc(S(N)(=O)=O)c1C 18011,N1(C(c2ccc(C#C)c(Cl)c2)=O)CC(NC(=O)C=CC2CC2)C2(CCOCC2)C1 18012,c1(NC(C2(C)CCN(C(C(C)(C)CCl)=O)CC2)=O)c(F)cccc1C#N 18013,Cc1cccc(C(O)C(=O)NC(C)CNC(=O)CC2CC3C=CC2CC3)c1F 18014,C1(NC(c2ccc(N(C)C)cn2)=O)CC2CCC1C(NC(=O)C1=CCCOC1)C2 18015,C1(CC(N2C(CCNC(=O)C(F)C3CCC3)COCC2)=O)CC(=O)NC(=O)C1 18016,c1(C(N2C(CNC(c3ccn(C)c3)=O)CCCCC2)=O)c[nH]c2cc(O)ccc12 18017,N1(C(c2c(CC)nco2)=O)CCC2(C1)CN(C(=O)C(C)NS(=O)(=O)CC)C2 18018,N1(C(c2cc(SC)c(C)o2)=O)CC(C)N(C(c2cn(C)c(C)cc2=O)=O)CC1C 18019,CCC1=NOC(C(=O)NCCCN(C(c2cnc(CC(C)(C)C)s2)=O)C(C)C)C1 18020,c1(C(C(=O)NCC(F)F)N(C2CC(=O)N(C)C2=O)C(C)C)cccc(C#N)n1 18021,C(=O)(CC1c2ccccc2CCN1S(C)(=O)=O)NCC1N(C(CC=C)=O)CC1 18022,N1(C(C2CCC(CC)CC2)=O)C(CNC(c2cc(Cl)cnn2)=O)CC2COCC12 18023,N1(C(c2ccc(C)cc2)=O)CC2(CC(NC(c3cnc(N)c(Br)c3)=O)C2)C1 18024,C1(Cn2cc(-c3c(CC)cccc3)nn2)CCN(C(=O)C(F)(F)Cl)CC1(F)F 18025,N1(C(Cc2ccc(C#C)cc2)=O)CCC2(CC1)CN(C(C1CCCS1)=O)C2C(C)C 18026,N1(C(C(COC)C)=O)CCOC2(CCN(C(C3CC(=O)C3)=O)C2)C1 18027,c1(C(=O)NCc2cc(C3CC3)ncn2)cccc(C2(F)COC2)c1.C1C(O)CN1 18028,CCCC(CCC)CC(=O)NCC1CN(C(c2cnn(CC)c2)=O)CCC1C 18029,n1(CC(=O)NC2C(CNC(c3cnc(C)s3)=O)C2)cc(Br)c(C)n1 18030,N1(C(C=NOC)=O)CC(CNC(=O)Cc2cccc(F)c2F)CC2(CCC2)C1 18031,CC1CCCn2cc(C(=O)NCC3CC3NC(C3CN(S(N)(=O)=O)C3)=O)nc21 18032,CCC(O)(C(=O)NCCCCC(C)NC(c1nc(C)cs1)=O)c1ccccc1 18033,N#CC1C2CCC1CN(C(C13CC(CO1)N(C(=O)CC1OCCO1)C3)=O)C2 18034,CN1CC(NC(C2CC23CC(NC(C2CCCCC2O)=O)C3)=O)C(C)(C)C1 18035,C1(C(N2CCCC(CN(C(=O)CC(C)(C)C)CC)C2)=O)CC12CCOCC2 18036,Cc1cc(Cl)cc(NC(C2CC(F)CN2Cc2ccc(C)c(C)c2)=O)c1O 18037,N1(C(C(C)OCC2CCCO2)=O)CCCN(C(=O)C(C2CCCCC2)F)CC1 18038,c1(C(N(CCCN(C(c2c(C)ccnc2)=O)C)C)=O)c(C)nc(O)nc1S 18039,n1(CC)nc(C(=O)NCC2CCC(NC(=O)CCCNC(=O)OC)C2)c(Br)n1 18040,c1(CC(N2C(CNC(C3(C#N)CCCO3)=O)CC(O)C2)=O)cc(F)ccc1Cl 18041,CC(C)CC(O)CNC(C1CCN(C2CCCN2NC(=O)Nc2ccccc2)C1)=O 18042,N1(CC)CCN(C(=O)CCC(=O)C(C)(C)C)C(=O)C12CCCC2 18043,N1(C(CC(C=C)CC)=O)CC2(C(=O)N(C)Cc3cncnc3)CC1CCO2 18044,c1(CC(=O)NCCC2(O)CCN(C(c3c(C)coc3C)=O)C2)cccc(Cl)c1Cl 18045,C1(C(N(CCNC(C(c2ccc(OC)cc2)CC)=O)C(C)C)=O)CSCC(=O)N1 18046,C1(N(C)C(C2CC=CCC2)=O)CCCN(C(c2conc2C2CCCC2)=O)C1 18047,c1(C(N2CC(CNC(C3CC(C(C)C)OCC3)=O)C2)=O)cc2nc[nH]c2cn1 18048,C(c1ccc(C)c(C)c1)=CC(=O)NCC(CCOC)NC(=O)C=CC(C)C 18049,c1(C(N(CC(C)N(C(C(CCC)CC)=O)C)C)=O)ccc2c(c1)CN(C)CC2 18050,C=CCC(C(=O)NCC1(CN(C)C(C2CCC3CC3CC2)=O)CC1)C(C)C 18051,C(=O)(C(C)(F)C(F)(F)F)NCC(C(C)C)(C)NC(C1CCN(C(N)=O)CC1)=O 18052,Cc1cc(Cl)cc(CNCC2OCCN(C)C2c2ccccc2)c1O 18053,C(C(CC(=O)NC1CCN(C(C2CCCS2)=O)CC1)C(F)F)N(C)C 18054,C1(NC(CCOc2c(CC)cccc2)=O)CCCCN(C(c2cnns2)=O)C1 18055,C=C(Cl)CC(C(=O)N1CCC1C)NC(c1nnn(CC)c1C)=O 18056,C(=O)(C(C)(C)C(=O)NC1CCCN(C(c2cscc2Br)=O)CC1)NC 18057,C1(NC(c2c(CC)oc(C)c2)=O)CN(C(c2cocn2)=O)CC12CC2 18058,C(=O)(C1=CSCCO1)N(CCN(C(C=C(CC)c1cccs1)=O)C)C(C)C 18059,N1(C(CN(c2ccncc2)C)=O)CCC2CC1CN2C(c1csc(Cl)c1)=O 18060,CC1CC(C)N(C(=O)C2=CCCSC2)CCN1C(c1ccc(Cl)c(C#N)c1)=O 18061,N1(C(C23CC(C)(C2)OC3(C)C)=O)CCC2CC(NC(c3cscn3)=O)CCC2C1 18062,C1(CCC(=O)N(CCOC)CCOC)CCN(C(=O)CN2C(=O)CNC2=O)CC1 18063,C1(NC(CCC#CC)=O)CCSC12CN(C(=O)CCOc1cccc(C)c1)C2 18064,C=CC1(C(N2CC(O)(c3cc[nH]n3)C2)=O)CCN(C(C2CC2C2CCC2)=O)CC1 18065,CC1(C)CC(SC(=O)NOCC(C2CCOC2)O)C1 18066,C1(C(=O)Nc2cn(C)nc2)C2CCC(F)C12.n12cc(nn1)CNC(=O)C2 18067,N1(CC(=O)NC2CN(C(C(C(C)C)F)=O)CC2C)CCc2ccccc21 18068,C12(NC(c3n(C)ccc3)=O)CN(C(=O)C(C3CCOCC3)O)CC1CS(=O)(=O)C2 18069,N1(C(c2ccc(NCC)cc2)=O)CCCC(F)(CNC(=O)CC2CC3(CC3)C2)C1 18070,Cc1ccc(NC(C2(CCNC(C34CC(C)(CCO3)C4)=O)CCC2)=O)cc1CO 18071,CCCCCCCC(=O)NCC(C)(O)CNC(C1CNC(=O)CC1(C)C)=O 18072,c1(C(=O)NC(C(=O)NC(c2cc[nH]n2)C)CC2CC2)cccc(F)c1N 18073,c1(C(N2CCCC(C)C2CNC(C2(N(C)C)CCC2)=O)=O)cccc2ccnn12 18074,Cc1oc2ccccc2c1C(N1CC(NC(C2CCCCS2)=O)CC1(C)C)=O 18075,C1(NC(=O)Cc2cncnc2)CN(C(=O)CCF)CCC1c1ccc(F)cc1 18076,c1(CCC(=O)NC(CNC(C(C)OC)=O)C)ccc(Br)nc1.C1C(=O)S1 18077,C1(C(=O)Nc2cccc(C(F)F)n2)CC(O)CCN1C(c1cccc(Cl)c1Cl)=O 18078,Cc1ccc(C(=O)NCC2CN(C(C3CN(C)CC(C)O3)=O)CC2C)nc1F 18079,CC1CN(C(=O)C(C)(C)C2CC2)CC2(CCN(C(c3cc(O)nc(O)c3)=O)C2)O1 18080,C(=O)(CC(C)C(F)F)N1CCC(CNC(CNC(c2c(C)occ2)=O)=O)C1 18081,Cc1ccc(C(F)(F)CNCc2nc(C3CC3)nn2C)c(C)c1 18082,C1(NC(CC(=C)I)=O)CC(C)CN(C(c2ccc(C)nc2)=O)C1 18083,c1(-c2cn(C3CCN(C(C4CCCO4)=O)C3)nn2)ccc(Cl)c(Cl)c1 18084,CC(C)(C)CCC(F)C(=O)N1CCC(CCC(=O)NCCOCCCF)C1 18085,C1(N(C)C(=O)NCCc2nc(-c3ccccc3)no2)CCCCC1C(F)(F)F 18086,C1(NC(CC2(OC)CCC2)=O)COC2(CCN(C(c3ccc(Cl)c(F)c3)=O)C2)C1 18087,CCC(C)(CO)C(=O)NC(C)CCCNC(=O)CCN1CCCCC1=O 18088,C1(C)(C(=O)NC(C=CC(=O)N(CC(=O)NC2CC2)CC)C)CC1(F)F 18089,C1(C(=O)NCc2ccc(-c3ccc(F)cc3)cc2)CCC2(CCCC2)C1 18090,C1(O)(C(=O)NC2CCC(NC(C3=NOC(C)C3)=O)CC2)CCCC(C)(C)CC1 18091,Cc1cc(C)c(NC(N2CCC(=CC(=O)Nc3cnc(OC)s3)CC2)=O)c(C)c1 18092,C1(CNC(C2(CC#C)CC=CCC2)=O)N(C(=O)Cc2cnsc2)CCC1(C)C 18093,C1(NC(C2(Cl)C(C)(C)C2)=O)CCCN(C(c2nc(=N)cc[nH]2)=O)C1 18094,c1(C(N2CCCC(C)(OC)C2)=O)cc2c(C)ccc(C)c2[nH]1.c12ccccc1OC2 18095,c1(C(C)=O)csc(C(=O)NCC2(O)CN(C(C3CC3(C)C)=O)C2)c1 18096,N1(C(CC(C)OC)=O)CC(C(=O)NCCNC(=O)C(C)C)C2CCCC12 18097,N1(C(C(=O)NC(C)C)=O)CC(NC(=O)C(c2ccccc2Cl)O)CC12CCC2 18098,C1(NC(C(C)=C2CCCC2)=O)CC(F)(F)CC1NC(c1ccc(CN(C)C)o1)=O 18099,c1(OC)cc(N(C)CCN(C)C(C2CCOC(C(C)C)C2)=O)nc(C(F)(F)F)n1 18100,c1(C(=O)NC2C(CNC(=O)CCC3CCCCO3)CCC2)cc(Cl)cnn1 18101,C1(NC(n2c(C)cnc2)=O)CN(C(C2CCCN2S(C)(=O)=O)=O)CC1C 18102,S(=O)(=O)(c1ccc(F)cc1)NCCC(=O)N(c1ccccc1)CC(C)C 18103,c1(NC(C2(SC)CN(C(c3cc(O)nc(O)n3)=O)C2)=O)cc(C)cnc1C 18104,c1(C(=O)NCC(CNC(CC(C=C)C)=O)OC)cc2cccnc2o1 18105,C1(NC(COCC(N2CCCC2)C)=O)CC2CC1N(C(c1cnnc(O)c1)=O)C2 18106,c1(NC(=O)NC23CC(NCc4ccc(C(=O)O)cc4Cl)(C2)C3)cccc(Br)c1Cl 18107,C(=O)(C(C)(C)CNC(=O)CC1CC=CCC1)N(C)CC1CCN(C)C1 18108,C(=O)(CC(C(F)F)NC(=O)CC1CCSC1)NCCCCC 18109,C(=O)(C1=CCCCO1)N1CC(NC(Cc2c(C)oc(-c3ccco3)n2)=O)C2C1C2 18110,CC1(C)CC(C(O)CNC(=O)CNC(c2cccs2)=O)C1 18111,C1(C(=O)NCCCC(C)NC(CCN(C(CCC)C)C)=O)CN(C(C)C)CCO1 18112,Cc1nc2c(Cl)cccc2cc1C(=O)NC(CNC(C1CNC(=O)N1)=O)C1CC1 18113,c1(NC(C(N2CCC(C(=O)OC)(C(=O)OC)C2)=O)=O)c(C)cc(Cl)nc1I 18114,C1(CC(=O)Nc2c(COC)n(C)nc2)CCCCC1(O)C(F)(F)F 18115,C1(NC(C2CCCC2)=O)CCOC12CCN(C(C1COC3COCC13)=O)CC2 18116,c1(C(=O)NCC(CNC(C(C=C)O)=O)CO)ccc2c(c1)OCCC2 18117,C1(CNC(C2N(CC)CCC2)=O)CCCN(C(=O)CCC(C)(C)N(C)C)CC1 18118,N1(C(C2CC(=O)NC2)=O)CCOCC(F)(CNC(C2CC2c2ccsc2)=O)C1 18119,c1(C(=O)NC(C(C)NC(CCN(C(CCC)C)C)=O)C)cc(C)nc(O)n1 18120,c1(OCCOC)ccc(C(=O)NCC(O)CNCc2nncn2C(C)C)cn1 18121,N1(C(CC(CNC(C(C(COC)C)C)=O)(C)C)=O)CCC2(CCOCC2)C1 18122,CCCCCCCCC(=O)N(C(CC(F)F)C(=O)NCC(c1cccnc1)O)C 18123,N1(C(c2sccc2Br)C(=O)NC(CC)C)CC(OC)CC(O)C1 18124,C(=O)(C1CCC(=O)c2cccn21)N1CCN(C(C2C(C)C2C)=O)C(CO)C1 18125,N1(C(=O)OC(C)(C)C)CCCCCC(NC(=O)NCC2CC23CC3)C1 18126,N(C(=NCCCP(C)(C)=O)NCC(C)SC)CC(c1cc(OC)cc(OC)c1)O 18127,C1(CNC(C2(OC)CCSCC2)=O)C2CCCC1N(C(c1nc(=O)n(C)[nH]1)=O)C2 18128,CN1CCC(C(=O)NC2(C)CC(NC(=O)C(F)CNC(=O)OC(C)(C)C)C2)CC1 18129,CC1CCC(C(=O)NCCC(C)(C)NC(c2ccc(Br)c(O)n2)=O)C(=O)N1 18130,N1(C(C(Cc2cc[nH]n2)NC(C2CN(C)C(=O)C2)=O)=O)CCN(C)C2(CCC2)C1 18131,c1(C(=O)NC2(CF)CN(C(C3OCC(C)C3)=O)C2)ccc(C#N)c(O)c1 18132,CCC(C(C)CN(C)C)NC(=O)C(Cc1cc[nH]n1)NC(=O)CCc1ccco1 18133,c1(C(=O)N(c2ncncc2I)CC2(F)CNC2)ccc(Cl)c(F)c1 18134,C(=O)(C(O)P(C)(C)=O)N1CCCC(NC(CS(N2CCC(C)CC2)(=O)=O)=O)C1 18135,c1(OC)c(C(=O)NC(C)CCCCNC(c2c(C)ncn2C)=O)cc(F)cc1F 18136,CC1(C)CC(NC(C2(C(N)=O)CC2)=O)Cc2ccccc21 18137,C1(C(C)NC(C(CC)N(C)C)=O)CCCN(CC(=O)Nc2cnccn2)C1 18138,N1(C(c2nc(CC)sc2)=O)CCCC(C)(CNC(=O)C=C(C)c2cccnc2)C1 18139,c1(SCCNC(N2C(c3scc(C(=O)OCC)n3)CCC2)=O)cccc(Cl)c1C 18140,c1(C(N2CC(NC(c3c(NC)nccc3)=O)C2)=O)ccc(-n2cncn2)cc1C 18141,N1(C(Cc2nc(C)sc2)=O)CC2(CNC(C3CCSC3)=O)CC1CO2 18142,O=C(C1=Cc2cc(Cl)ccc2OC1)NC1C2CC1N(C(=O)COC(F)(F)F)C2 18143,CC(C)C(C(=O)NC(C1(C)CN(C(=O)C(=O)NCC2CC2)C(C)(C)C1)C)C(C)C 18144,C1(NC(N2CC(COC)C(CC(C)(C)C)C2)=O)CCC(OC)CC1OC 18145,C(=O)(C(C)CC(F)F)N1C(C=CC(=O)N(CC)Cc2cn(C)nn2)CCC1 18146,C1(C(=O)NCCc2cc(C(=O)NCC3CCSC3)no2)C2CCC(=O)C12 18147,N1(C(c2c(OCC)scc2)=O)CCC2(CCCN(C(C3COC(=O)C3)=O)C2)C1 18148,C(C(C)(O)C(C)CC)NC(CC1CCC(NC(C2(CC=C)CC2)=O)CC1)=O 18149,Cc1ncsc1C(=O)NCC(O)CN(C(C1CCC1c1ccccc1)=O)C(C)C 18150,C1(C(C)O)CCN(C(=O)C(=O)N(Cc2ccccc2)CC2CCOCC2)C1 18151,c1(C(N2CC(CCCCNC(CCC=C)=O)C2)=O)nnn(CCOC)c1N 18152,c1(C(=O)NC(CC(C)NC(CNC(=O)NC)=O)C)cc(C(C)C)ccc1F 18153,CN1C2CC(O)C1CC(c1nnnn1C)(NCc1cnn(CCF)c1)C2 18154,N1(C(COCC(=C)C)=O)CC=CCC1C(=O)NC1CC(C)OC1=O 18155,C(=O)(CC(O)C(C)CC)NC1(CC=C)CCN(C(C2(Cl)CC2)=O)CC1 18156,C(=O)(CC(CNC(=O)C(C(C)C)NC(=O)N(C)C)c1ccc(Cl)cc1)OC 18157,n1(CC)nncc1C(=O)NC(C)C=CC(N1CCC(N(C)C)C1)=O 18158,c1(C(=O)NCCC2CCN(C(C3C(C=C)C3)=O)C2)c(-n2cccc2)sc(C)c1C 18159,C1(S(C)(=O)=O)(CNC(c2c(SC)cc(Br)cc2)c2nnnn2C(C)C)CCCC1 18160,OCCC#CCN=c1ccnc(NCCn2cc(Br)ccc2=O)[nH]1 18161,N(C(=NCCC)NCC1CC1C1CCCO1)CC1C(c2cccc(OC)c2)C1 18162,c1(C(C(F)(F)F)OC(=O)Cn2cnc(Br)n2)ccc(OCC(F)F)nc1 18163,c1(CC)nc(C(=O)N(CC(N2C(CO)CC2C)=O)CC2CC2)co1 18164,N1(C(c2c(COC)cco2)=O)CC2CC1CN2C(c1cc(C(C)C)on1)=O 18165,CC1CN(C(C2CCCC2CNC(C2CC(O)CN2C)=O)=O)CCS1 18166,Cc1nc(Cl)ccc1CC(N1CC(OC2CCN(C(=O)C(C)C3CC3)CC2)C1)=O 18167,c1(C(=O)NC(CCOC)CNC(C2CN(C)C(=O)N2)=O)cc2[nH]ccc2s1 18168,C1(CNC(c2c(C)coc2C)=O)CC(C)(C)CCC1NC(=O)CC1CC(F)(F)C1 18169,c1(C(=O)NC2(CO)CCCN(Cc3ccccc3)C2)cccc([N+](=O)[O-])c1O 18170,C1(NC(C(C(C)C)SC)=O)CCN(C(=O)CC2CCCCC2C)CC1F 18171,C1(NC(c2ccc(CC)[nH]2)=O)CCCC(CNC(c2cn(C3CC3)nn2)=O)C1 18172,N1(C(COCCOC)=O)CC=C(C(=O)NC2(CO)CCOC2)C1 18173,C(C(C)(C)CNC(c1ccc(CNC(=O)CSCCC(F)(F)F)o1)=O)N(C)C 18174,C1(C(=O)NC2CC(N(C(c3ncn(CC)c3)=O)C)C2)CC(C(C)C)=NO1 18175,c1(C(N(c2ccccc2)CCCC)=O)cc(F)c(Br)cc1F 18176,O=S(=O)(c1[nH]c(=NCC(O)c2cccnc2)ccc1Br)NC1CC2(CCC2)C1 18177,N1(C(C#CC(C)C)=O)CC2CCOCC2(NC(=O)COc2ccc(Cl)cc2)C1 18178,C(=O)(CCCC(C)(C)C)N(C1CCN(CCC2CCCCO2)CC1)CCC 18179,C1(NC(c2ccc(OCCCOC)cc2)C)CCCC(C)(C)C1 18180,c1(C(=O)NC(CCC)CNC(c2cnc(C3CC3)s2)=O)cncc(Cl)c1 18181,C1(NC(C2C=C(C)CS2)=O)CCC(C)(CNC(=O)Cc2csnn2)CC1 18182,N1(C(c2nccc(C(F)F)n2)=O)CCCCC2(CCN(C(C3CC3(Cl)Cl)=O)C2)C1 18183,c1(C(N2CCC(NC(COCCC(C)C)=O)(CF)C2)=O)nnn2c1CCCC2 18184,CCC(C)(CCC(C)C)C(=O)N1CC(NC(=O)CCc2cnn(C)n2)C2(CC2)C1 18185,c1(C(N(C2CCCN(C(C3(N(C)C)CCSC3)=O)C2)CCC)=O)ccccc1C 18186,C1(NC(C(CN(C)C)CO)=O)CCC2(CCN(C(=O)CCOC3COC3)C2)C1 18187,N1(C(CCCNC(c2cnn(C(F)F)c2)=O)=O)CCCC2CCCC12 18188,CC1(C)CC(C(=O)NC2CC2NC(c2cnc(-c3cccs3)s2)=O)=NO1 18189,c1(C(N2CCCC(NC(c3cncc(C#C)c3)=O)CC2)=O)c(C)nc(O)nc1S 18190,c1(OC)ccc(C(N2CC(CN(C)C(C3CCC(O)CC3)=O)C2)=O)c(N)c1F 18191,N1(C(c2cc(CC)ncn2)=O)CCCC(C)C1CCNC(=O)CN1CC2CC2C1 18192,O=C(NOCCc1ccccc1)C(=O)NC1(C(=O)O)CCOCC1 18193,CCCC(CC)CCC(=O)N(C)CC1(O)CCN(C(c2cc(F)cc(Cl)c2)=O)C1 18194,C(c1ccncc1C)=CC(N1CCC(NC(c2ccn(C(CC)CC)n2)=O)C1)=O 18195,C1(NC(C(c2ccc(C)cc2)(C)C)=O)CCCN(C(c2ccc(C#N)s2)=O)C1C 18196,c1(N2C3(CN(C(c4c(OC)ccs4)=O)C3)CCC2)ccnc(S(=O)(=O)C(C)C)n1 18197,Cc1cc(C(=O)OCc2cnoc2C2CC2)nnc1C 18198,C1(c2ccccc2)(CNC(CC=C)=O)CCN(C(c2coc(O)n2)=O)CC1 18199,N1(C(Cc2nnc(C)o2)=O)CCC(CNC(=O)Cc2cnsc2)C12CCC2 18200,N1(C(c2cc(F)cc(Br)c2F)=O)CCN(Cc2cscn2)CC12CC2 18201,C1(C(N2C(c3cccc(C)c3)C(=O)NCC2)=O)COc2cc(F)ccc2C1 18202,N1(C(c2n(C)c(O)nc2)=O)CC(NC(C2CC2c2ccc(Cl)s2)=O)CCC(O)C1 18203,CCC(CCCC(=O)NOCc1ccccc1)NC(C1CC2(CC2)C1)=O 18204,Cc1csc2ncc(C(=O)NCC3CCCN(C(C4CNC(=O)C4)=O)C3)c(=O)n12 18205,C1(N(C(C)=O)C)CCCCC12CCCN(C(=O)C1CC1)C2 18206,c1(CCC(N2CC3(CN(Cc4cncc(C)n4)C3)C2)=O)c[nH]c2ccc(F)cc12 18207,C(CC(=O)NC1(C)CCCC1(C)C)(C(C)OC)NC(CCCC)=O 18208,c1(CC)oc(C)cc1C(=O)OCc1ccnn1C(F)(F)F 18209,N1(C(CN(S(CC)(=O)=O)C)=O)CCC2(CC1)CC2CNC(=O)CC(C)CN(C)C 18210,CC1C(=O)N(C)CCN1Cc1nc(-c2sccc2CO)cs1 18211,N1(C(CN2C(C)CCCC2)=O)CCC(NC(=O)CC2CCC(=O)NC2)C(C)(C)C1 18212,N#Cc1cc(N2CCCC2CNC(c2cccc3c2ncn3C)=O)ccc1[N+](=O)[O-] 18213,C=C(C)CCC(=O)NC1CCCC1NC(=O)CCC(=O)c1ccccn1 18214,c1(C(N2CC(C)N(C(=O)CC3CCC4CC4C3)CC2)=O)cc2ncccc2[nH]1 18215,C1(C(=O)NCC(C)(C)NC(Cc2c(C)noc2)=O)CCS(=O)(=O)C1 18216,C1(NC(C(=O)OCC)=O)CCC(CCC(=O)NCCNC(N2CCCC2)=O)C1 18217,C1(CCOC)CN(C(C2CCCN2C)=O)CCN1C(=O)CP(C)(C)=O 18218,N1(CC(C(C)(C)C)=O)CC2(CCC(CNC(C3CCCCO3)=O)O2)C1 18219,C1(OC)(CNC(C2(c3cc[nH]n3)CC2)=O)CCN(C(C2CC(=O)N(C)C2)=O)CC1 18220,c1(CC)cc(F)ccc1CC(N1CCC(NC(=O)COC(C)CC)C1C)=O 18221,N1(C(CC=CCCCCC)=O)CCN(C(=O)CN=S(C)(C)=O)CC(C)C1 18222,C(=O)(NNC(=O)C(C)(C)CCCCNC(c1cccnc1)=O)c1c(C)ccs1 18223,n1(CCNC(C(C)c2ccco2)=O)cc(C(=O)NCC(C)OC(F)F)cn1 18224,CC1(C)C(C)(C)C1(F)CNC(=O)CNc1cnc(Cl)c(Cl)c1 18225,C1(NC(C(C)(C)c2cccs2)=O)CCN(C(=O)C=C(Cl)Cl)CC1O 18226,N1(Cc2cc(C)c(F)cc2)CCC(F)(F)C(C(=O)NCc2ccsc2Br)C1 18227,c1(OC)ccccc1C(=O)C(=O)NC1CC(C)N(C(=O)CCc2cnc[nH]2)C1 18228,C1(C(N(CC(C)(C)NC(=O)CC(F)(F)Cl)C)=O)CCCC1S(C)(=O)=O 18229,c1(C(=O)NCCCNC(=O)COCCOCCCNS(CC)(=O)=O)ccc(O)nc1 18230,c1(NC(=O)CC2COCCN2Cc2c(C)n[nH]c2)ncc(Br)c(C)c1[N+](=O)[O-] 18231,N1(C(C(=O)NCCc2c(Cl)cccc2Cl)=O)CCC2(CC(=O)NC2=O)C1 18232,c1(CC(=O)NC2C=CCN(C(C(C)Oc3ccccn3)=O)C2)c(Cl)cccc1Cl 18233,N1(C(CCSCCC)=O)CCN(C(c2ccc(CC)cc2)=O)C2CCCCC2C1 18234,C1(C(=O)NCC2C(CNC(Cc3c(C)cnn3C)=O)C2)CC2CC(=O)C1C2 18235,C1(C(N(CC)CC2CCCN2C(=O)CC#N)=O)Cc2cccc(F)c2O1 18236,N1(S(c2cn(CC)nc2C(F)(F)F)(=O)=O)CCC(CN)c2ccccc21 18237,C1(CC)CCN(C(=O)CC2CN(C(c3cc(C)[nH]n3)=O)C2)C1CNC(C)=O 18238,c1(CC(=O)NC(CC)CNC(C2(C)C=CCC2)=O)ccc(OC)cc1Br 18239,C(=O)(CC(C)C(=O)N(CC(C1CC1)OCC)C)OCC.C1C(=O)N1 18240,Cc1cc(Br)cnc1C(c1nnnn1C1COC1)NCCC1CCC(C)(C)C1 18241,CCC(C(O)C(F)(F)F)NC(=O)NC(c1ccccc1)CF 18242,S(=O)(=O)(CC(=O)NC1COCC1CNC(c1c[nH]nc1OC)=O)N(CC)CC 18243,Cc1ncc(C=CC(=O)NCC2CCN(C(C3(O)CCOC3)=O)C2)c(O)n1 18244,c1(C(=O)NCC(C2CCOC2)NC(Cc2nc(C)[nH]n2)=O)nc(O)c(C)s1 18245,N1(C(c2cn(C3CCN(C)C3)nn2)=O)CCCC(CN(C(=O)CC(F)F)C)C1 18246,N1(C(C(N2CCCCC2=O)C)=O)CCC2(CC1)CC(NC(=O)CC(C)(C)C1CC1)C2 18247,c1(CC)ncc(Br)c(C(=O)NC2C3CN(C(=O)Cc4[nH]cnc4C)CC23)n1 18248,Cc1cccc2c(C(N3CC(C)(C)CC3CNC(=O)C(C)CO)=O)nccc12 18249,C=CC1(C(=O)NC2(C(=O)OC)CC2)CCN(C(C2CC=CC2)=O)CC1 18250,C=CCC(CO)NC(=O)COCCNC(C1CC12CC2)=O 18251,C1(NC(C(C)Oc2cccnc2)=O)CC(C)N(C(=O)CCC2CC2(F)F)C1 18252,c1(NC(C)=O)cnccc1C(=O)NCC(C)CN(C)C(c1conc1C)=O 18253,c1(CC#N)cccc(C(N2CC=CC(NC(=O)CCC3CC3(F)F)C2)=O)c1 18254,c1(OCC)cc(C(N2CCC(CNC(=O)C3=CCC(C)CC3)C2)=O)cc(Cl)c1O 18255,C1(NC(c2cc(C)c(O)nc2)=O)CC2CCC(C1)N2C(C1(n2cccn2)CC1)=O 18256,CCCCCC(CC)C(=O)N1CCC(CNC(=O)CCC2CC2)(COC)CC1 18257,N1(C(CCc2cncc(C)c2)=O)CC2CN(C(c3ccc(C)nn3)=O)CCC12 18258,C(=O)(CC(C(C)OC)NC(c1ccc(O)cc1F)=O)NCCCCCC=C 18259,c1(CN2CC3C(C(=O)NCc4ccc(F)cn4)C3C2)cccc(O)c1F 18260,C1(C(=O)NCC2N(C(c3c(C)cc(C)s3)=O)CCC2)CCC(=O)CC1(C)C 18261,N1(C(CC2C(C)OCC2)=O)CCC(C(=O)NCc2cnn(C)c2)C12CCC2 18262,c1(C(N(C2CC(NC(C3(C)CS(=O)(=O)C3)=O)C2)C)=O)cc2c(cc1O)CCCC2 18263,c1(OCC)ncc(C(=O)NC2CC(CNC(c3ncn(C)n3)=O)C(O)C2)cn1 18264,Cc1cc(C(C)C(=O)NC2CCCN(C(C3CCCO3)=O)C2)cc(F)c1 18265,C(=O)(C(C)P(C)(C)=O)N(CCOC)CCNC(=O)Cc1c[nH]ccc1=O 18266,CC1CCN(C(c2scnc2C2CC2)=O)CC1CNC(=O)C=Cc1ccsc1 18267,C(CCCCCN=[N+]=[N-])N(CCNc1ncccn1)C 18268,C(=O)(CCC(F)(F)C(F)F)OCC1C2N(C(=O)OC(C)(C)C)CC(CC2)C1 18269,Cc1ncc(C(N2CCC23CN(C(c2cn4ccnc4s2)=O)C3)=O)c(C)n1 18270,C1(C(=O)NCC(CNC(c2cc(-c3nc(C)sc3)oc2)=O)O)CCCCC12CC2 18271,N1(C(c2c(CC)ncs2)=O)CCOC2CCN(C(=O)C(C)c3ccsc3)CC12 18272,c1(C(=O)NCCN(C(CC(C)OC)=O)CCCN(C)C)csc(C)c1C 18273,c1(C(=O)NCCCN(C)C(c2cccc3ccoc23)=O)cc(F)c(O)c(Cl)c1 18274,c1(C(CC)=O)cc(C(N2CCC(CCNC(C3CC4CC3C4)=O)C2)=O)ccc1F 18275,c1(OCC(C)O)ccccc1NC(=O)NCC1CCCC(C(F)(F)F)C1 18276,n1(C(C)C)cc(C(N2CC(NC(c3cc(C(N4CCCC4)=O)c[nH]3)=O)C2)=O)nn1 18277,C1(O)(CNC(c2ccc(C(F)F)nc2O)=O)CCCN(C(C2(F)CCOC2)=O)C1 18278,C1(C(=O)NC2CC2CCCN(C(COC(CC)C)=O)C(C)C)CCN(C)CC1 18279,C1(NC(CCOCCC)=O)COC2(CCN(C(=O)CN3CCOCC3)C2)C1 18280,Cc1ccc(C(=O)NC2CC3CN(C(C4(F)CCCC4)=O)CC23)c(C(C)C)n1 18281,C(=O)(CCCCCC#N)N1C(C)(C)CC(NC(C2CC23CCC3)=O)C1 18282,c1(C(=O)NCCCCC2CN(c3c(C)cnc(C)n3)C2)cc(C)c(C)cc1Cl 18283,c1(C(N2C(CCNC(C3CCC(=C)CC3)=O)CCC2)=O)ccc2nc(S)oc2c1 18284,N1(C(c2ccccc2Oc2cccnc2)=O)CCN(C(C2CC2F)=O)C(CF)C1 18285,c1(C(=O)NC(C(C)NC(C2(CC)COC2)=O)C)cccc(P(C)(C)=O)c1 18286,C1(C(=O)NC(CC=C)CO)CN(Cc2ccccc2C(=O)O)CCS1 18287,c1(C(=O)NCCOCCCNC(C2(C)CC2(F)F)=O)cc2ccncc2s1 18288,N1(C(CCc2cn(C)nc2)=O)CCN(C(=O)CSc2cnn(C)c2)CC12CCC2 18289,N1(C(C2(CC)CC2(F)F)=O)CCC(C2(NC(C3CCCCCC3)=O)CC2)C1 18290,c1(C(N2CC3C(NC(=O)C4=CCCC4)C3C2)=O)ccc2c(c1)C(=O)NCCO2 18291,N1(C(C(C)O)=O)CC2(CC2C(=O)Nc2ccc(N3CCCCC3)nc2)C1 18292,C1(CC(N2C(C(N)=O)CCC2)=O)CN(NC(C2CC3(CC3)C2)=O)CCO1 18293,N1(C2CN(CC(=O)N(C(c3nnnn3C(C)C)C)C)C2)CC(C(=O)N(C)C)CC1=O 18294,c1(C(=O)NC2C(CC)N(C(=O)C(CC)(CC)OC)CC2)cncc(F)c1C 18295,C1(CN(C(c2c(OC)csc2)=O)C)COCCN1C(=O)CCCc1n[nH]c(=N)s1 18296,N1(C(C23CC(NC(C(C)(CO)OC)=O)(C2)C3)=O)CCCC(C)(C#N)C1 18297,S(=O)(=O)(c1cccc(Br)c1)NC1CCN(C(c2sc(Cl)nc2Cl)=O)C1 18298,c1(OC)cc(CN2CC3CCC2CN3C(c2c(O)cccc2F)=O)cc(F)c1O 18299,CCC(O)C(C)(C)C(=O)NOCC(N1CC2CCC2(C(=O)OC)C1)=O 18300,C1(CC)CNC(=O)CN1C(C1CC=CCN1C(=O)C(C)NC(C)(C)CC)=O 18301,N1(C(C2C(C)OC(=O)N2)=O)CC2CN(C(C3CCC3)=O)CC2(C(F)(F)F)C1 18302,c1(C(N(C2CCN(C(C3CCC3(F)F)=O)C2)CCC)=O)ccnn1CC 18303,CCC(C)(C)C(O)C(=O)NCCCN(C)C(C1CC1c1ccoc1C)=O 18304,c1(C(C)C)nocc1C(=O)NC1CCN(Cc2nnn(C)n2)C1 18305,C(=O)(C(CCCC)NC(=O)C(C)SC(C)C)NC(c1cccnc1)C#C 18306,C1(O)(C(=O)NCCC2(C(=O)OC)CCCC2)CCNCC1 18307,C1(NC(C2(C#N)CCC2)=O)CCC(NC(=O)CN2CCOCC2)CC1 18308,Cc1nn(C)c(Cl)c1C=CC(N1CC(CNC(=O)Cn2ccc(O)nc2=O)C1)=O 18309,N1(C(C2(NC(c3n[nH]c(O)n3)=O)CSC2)=O)CC2(C1)NC(=O)NC2=O 18310,c1(OC)cccc(C2CC2C(=O)NCCC2CCCN2C(C2CC(Cl)(Cl)C2)=O)c1 18311,C1(CNC(CCCOCCC)=O)CCCC(NC(=O)CCC=CBr)C1 18312,CC(CC(F)F)C(=O)NC1CN(C(c2ccsc2)=O)CC12CC2 18313,c1(CCNC(C(c2c(CC)noc2)N(CC#N)CCOC)=O)ccccc1F 18314,c1(C(=O)NCCC(C)NC(C2(COC)CCOCC2)=O)ccc2nc(C)sc2c1 18315,C1(C(=O)NC2CC(CC(=O)NCC(C)OCC=C)C2)CCCC(=O)N1 18316,C1(NC(c2n(CC)ncn2)=O)CCC2CN(C(c3nccnc3N)=O)CC2C1 18317,c1(NC(c2ccc(CCNC(CCCC=C)=O)cc2)=O)ccc2nnsc2c1 18318,CC(C)CC(CC(C)C)C(=O)NC1CC1NC(C1(Cl)CC1)=O 18319,N#Cc1cc(F)ccc1C(=O)NCC1CN(C(c2cc(Cl)cc(Cl)c2Cl)=O)C1 18320,CC1C(C)N(C)CCN1C(=O)C#CCNC(C1COCCN1C)=O 18321,Cc1c(C(N2CC(=O)CC2C(=O)NC(CC2CC2)C2CC2)=O)nnn1C 18322,N1(C(C(C(C)C)=O)=O)CCN(C(c2cnccn2)=O)C(C)C1 18323,C(=O)(CC(O)CC(C)(C)C)NCC1N(C(c2nc(OCC)sn2)=O)CC=C1 18324,N1(C(=O)NCC2(OC)CC2)CCC(O)C(C(=O)NCCC(C)OC)C1 18325,c1(C(=O)NC2CC(C)(NC(=O)CC3CC34CC4)C2)csc2c1CCCC2 18326,Cc1nc(NCC2CCC(C)(C)CC2)cc(=NCc2cc(Br)cs2)[nH]1 18327,c1(OC)nc(C)ccc1C(=O)NC1CN(C(c2cnc(O)nc2O)=O)CC12CC2 18328,C(CCC(C)(C)C(=O)N(CC(C1CC1)OC)C)NC(c1ncc(CC)cn1)=O 18329,c1(C(N(C2CCCN(C(=O)Cc3cnns3)C2)C)=O)cnc2c(c1)NCC2 18330,C(C1CN(C(C2CC2c2ccco2)=O)CC1C(=O)NC1CC(C)C1)=CC 18331,N1(C(CC(C)SC)=O)CC(C)(C)CC1CNC(=O)CC1CCS(=O)(=O)C1 18332,N1(C(c2c(C)nco2)=O)CC(C)(C)OCC1CNC(C1(C)CC2CCC1O2)=O 18333,C1(C)(COC)CCCN1C(=O)CONC(c1nnn(CC)c1C)=O 18334,CC1CN(C(=O)C(C)(C)C)CC1CCNC(C1(C#N)CCC1)=O 18335,CC(CO)C(C)N=c1[nH]c2cc(Cl)c(S(=O)(=O)NCCC3(C)CCCC3)cc2s1 18336,C1(C(C2CCOC2)NC(CSS(C)(=O)=O)=O)CCCN1C(=O)CC1CC=CC1 18337,C1(=O)CC(CC(C)C)CN1.CCCCCCCC1CCCN1C(=O)C(F)(F)F 18338,c1(CC(=O)NCCN(C(c2sccc2C#N)=O)CC)cc(F)ccc1OC 18339,C(=O)(C#CC1CCCC1)N(CCCNC(c1c(C)cnn1C(C)C)=O)C1CC1 18340,CC1(C(=O)NC2CCCCC2NC(c2cc(N)cc(O)n2)=O)CCC(=O)NC1 18341,N1(C(C)C)CCCC(CC(=O)N(C2CCCN(C(c3cncc(F)c3)=O)C2)C)C1 18342,N1(C(=O)NC(CN(C)C)C(=O)N2CCOCC2)CCOC(c2nn[nH]n2)C1 18343,C(=O)(CS(=O)(=O)CC(C)C)NCC1(O)CN(C(c2cnc(C)[nH]2)=O)C1 18344,CC(C)(CC(=O)NC1CCCN(C(c2nccc3c[nH]nc23)=O)C1)CC(F)(F)F 18345,CCC(C(=O)N1CC2CC2(CNC(C2CN(C3CCC3)C2)=O)C1)C(F)(F)F 18346,CC(CCN(C(=O)CC1CCCO1)C)NC(=O)C=C1CCC1 18347,CCC(CC)(CO)C(=O)N1CCC(O)C(NC(=O)C=CC2CCC2)C1 18348,CC(C)CC(O)C(C)C(=O)N1CC(C(=O)NCC2(C)CCOCC2)C(C(C)C)C1 18349,N1(CCNC(CC(C=C)C)=O)CCN(C(=O)CC2CCC(C)(C)C2)CC12CCC2 18350,Cc1nn2ncccc2c1C(=O)NCC1CCCCN1C(c1ccncc1Cl)=O 18351,CC(C)(C)CC(C)(C)C(=O)NCc1csc(C(=O)NC2CCCC3(CC2)CC3)c1 18352,CN1CCOC(C(=O)NCCCCCCNC(=O)COC(F)F)C1 18353,c1(C(C(=O)NCCC2(O)CN(C(C(C)SCC)=O)C2)C)ccc(F)c(F)c1 18354,c1(N2CCN(CC)CC2)ccccc1C#N.C(CCC(C)N)N(CCO)CC 18355,c1(CNC(C2(F)CCN(C(C=Cc3cn(C)nc3)=O)C2)=O)nnc2n1CCC2 18356,C=CCC(C)(C)CC(=O)N1CCC(C)C(CNC(=O)C(CC)C(=O)OCC)C1 18357,c1(C(N(CCNC(=O)C(C2(O)CCCCC2)(F)F)CC)=O)cnc2nccn2c1 18358,N1(C(CC2CC(OC)C2)=O)CCN(CCN(C)C(C2CCCS2(=O)=O)=O)CC1 18359,C(CCN=C(NCc1ccc(CO)nc1)N1CCC(F)(c2ccccc2)C1)OC 18360,c1(C(=O)NCCCN(C(C(CC(C)C)(F)F)=O)C)cc(=O)c2ccccc2o1 18361,c1(C(=O)NCC2N(C(CNS(C)(=O)=O)=O)CC(F)C2)c(OC(F)F)cccc1F 18362,c1(OCCOC)cc(OC(C23CN(C(=O)OC(C)(C)C)C(C)(C2)C3)=O)ccc1O 18363,c1(C(=O)NCC(C)NC(c2snc(O)c2Cl)=O)ccc(C2COC2)cc1 18364,C1(NC(N(CC2=CCSC2)C)=O)CCCC1(C)CN(C)C 18365,n1(CC)ccc(C(=O)NC(CNC(=O)C(C)n2cnnn2)CO)n1 18366,C1(CNC(c2cscn2)=O)CN(C(C2C3CCC2CC3)=O)C2(CCOCC2)C1 18367,c1(OC)cccc2cc(C(C)NC(=O)NCc3ccc(C#N)c(OC)c3)oc12 18368,c1(C(=O)NC(C(C)NC(=O)CCC2CC2)(C)C)cc2ccccc2n1C 18369,CCCCCC(C)CC(=O)NC(C(=O)NCC1(CN=[N+]=[N-])CC1)C(C)(C)C 18370,C(=O)(CC(C)CC(C)(C)C)N1CCC(C(=O)NC(c2nccs2)CC)(SC)C1 18371,Cc1cc(CNC(=O)C(C)(C)C2CCCN2C(=O)CC(C)N(C)C)ccc1F 18372,c1(CC)cccc(-n2cc(CCC3CN(C(c4cnc(Cl)n4C)=O)C3)nn2)c1 18373,CCC(C)(C)C(O)C(=O)N1CC(F)CC1CN(C(=O)C(C)C)C 18374,CC1CN(C(C2CC(O)CN2C(c2ccc(CO)s2)=O)=O)CCC1N(C)C 18375,CC1CCCN(C(=NCC(O)C2CC(F)(F)C2)NCc2cccs2)C1 18376,N1(C(COc2c(OCC)cccc2)=O)CCC(C)(C(=O)N(C)CC#N)C1 18377,c1(OC)ccc2[nH]cc(C(N3CCC4CCC(C3)N4C(=O)CO)=O)c2c1 18378,c1(C(N2CCC(CC(=O)Nc3c(C)c(I)ccc3)C2)=O)cccn2cncc12 18379,C(=O)(CCCCCNC(N)=O)NC(C)CNC(=O)Cn1cc(C(C)O)nn1 18380,Cc1cncc(CC(=O)NC23COC(CNC(c4cc(CO)c(C)o4)=O)(C2)C3)c1 18381,Cn1c(O)nc2c(C(N3CC4CCN(C(=O)CC5CSC5)C(C4)C3)=O)cccc12 18382,C1(NC(C2(C)CNC(=O)C2)=O)CCCCN(C(C2CC2(F)F)=O)C1 18383,c1(C(N2CCC(NC(c3cc(C(=O)OC)on3)=O)CC2)=O)cncc2cnccc12 18384,C1(N(CCC)C(C2CCCC2O)=O)CCN(C(=O)CC2CCSCC2)CC1 18385,N1(C(c2cn(CCCC)nn2)=O)CC2CC1C2NC(c1snnc1CC)=O 18386,Cc1cc(CCCNC(=O)C(C)Sc2ccccn2)oc1C(=O)O 18387,c1(C(N(CCN(C(CC(CC)OC)=O)C)C)=O)[nH]cc2c1CCS2(=O)=O 18388,Cc1cccc(C(=O)NCCC2(O)CN(C(=O)CCOc3cccnc3)C2)c1 18389,C1(NC(C2CCC(C)(C)O2)=O)CN(C(=O)C=Cc2cc[nH]n2)Cc2nccn2C1 18390,C=CCCC(C(=O)OC)NC(=O)C(C)CN(C(=O)C(C)CC(N)=O)C 18391,c1(C2C(C)C2)ccc(CCC(=O)N(C)CCN(C)C(c2coc(Cl)c2)=O)o1 18392,C(CC(=O)N(CC(C)CC)C)(C(F)(F)F)NC(C(CC#C)C1CC1)=O 18393,c1(C(C(=O)NCCOC2CN(C(COCCOCC)=O)C2)(C)C)cccc(C#N)c1 18394,c1(OC)c(F)c(NC(=O)C(N2CCN3CCC2C3)=O)cc(F)c1F 18395,c1(C(N2CC(C)C(NC(=O)CCOC3CCC3)C2)=O)cc(F)ccc1Br 18396,CC1CC(c2nnnn2C)(Nc2ccc(Cl)c(Cl)c2)CC(C)O1 18397,C(c1ccncc1C)=C(CC)C=CC(=O)NCc1ncoc1C1CN(C(C)=O)C1 18398,CC1(C)C2CCC(C(=O)NC3CC3NC(C3C4CCCCC34)=O)C1C2 18399,C1(C(=O)NC2CC(C(N(c3cn(CC)nc3)C)=O)C2)C2CCCC(=O)C12 18400,C12(CNC(c3cnc(C4CCCCC4)s3)=O)CC(CO1)N(C(=O)C1CC1)C2 18401,C1(CONC(c2ccn(C)n2)=O)CC(C(N)=O)=NO1.N12CSCC1C2=O 18402,c1(C(N2C(CNC(C3C(C4C(C)C4)C3)=O)CC2)=O)cnn2cc(C#N)cnc12 18403,CC(C)(CNC(=O)Cn1cc(Cl)cn1)C(=O)N1CC2C=CC2C1 18404,c1(CC(=O)NC2CC(F)CN(C(c3c[nH]ccc3=O)=O)C2)cccc2sccc12 18405,CC(C)C(C(=O)N(CC(=O)NCCC12CCCC1C2)C1CCC1)C1CC1 18406,c1(NC(N(C(CCCSC)OC)C)=O)nc2ccccc2c(Cl)c1Br 18407,c1(-c2onc(C3N(C)CCNC3)n2)ccnc2[nH]ccc12 18408,c1(C(=O)NCCCCCNC(CCCC(=O)NC(C)C)=O)ccnc2c1CCO2 18409,C(=O)(C(C)(C)C(F)F)N(c1cn(CC(O)(C(F)(F)F)c2ccc(Cl)cc2)nn1)C 18410,C1(NC(CCC2CC(C)C2)=O)CCCC1NC(c1ccc(Cl)s1)=O 18411,O=C(C1=NOC2COCC12)OCCOc1cccc2ccccc12 18412,C1(C#N)(C(=O)NCC(CNC(=O)C(C(C)C)N(C2CC2)CC)OC)CC1(C)C 18413,N1(C(c2c(C)nco2)=O)CCOC2(C1)CN(C(c1cc3c(C)n[nH]c3cn1)=O)C2 18414,C1(C(=O)NCCCN2CCC(NC(C3CS(=O)(=O)C3)=O)CC2)CCc2nncn2C1 18415,CP(C)(=O)c1cccc(C(=O)NCC2CCC2NC(C2CC3CCC3C2)=O)c1 18416,c1(C(N(C(c2ccc(Cl)cn2)C)C)=O)cc(C(F)(F)F)ccc1F 18417,Cc1nc2nccc(C(N3CC(N(C(=O)CC4CC(F)(F)C4)C)C3)=O)n2n1 18418,C1(C(N2C(CCNC(C(COC)O)=O)CCC2)=O)CN2CCN1CC2C 18419,N1(C(C=C(CCC)C)=O)CC(C2CC2)(C(=O)NCCCCC2CC2C)C1 18420,c1(C(=O)NCCC(Cc2ccccc2)NC(CCC)=O)sc2cncn2c1C 18421,C=CC1(CC(=O)NC2CCCC(O)C2)CN(C(c2cocc2CC)=O)C1 18422,S(=O)(=O)(c1c(OC)ccc(Br)c1F)N(CCN(C)C)CC 18423,C12(C(N3CC(C)(NC(CC(CC)C4CC4)=O)C3)=O)CCCC(C1)OC2 18424,n1(CC(=O)N(C2CN(C(C3C(C(C)C)C3)=O)C2)C)cc(S(N)(=O)=O)cn1 18425,c1(C(=O)NC(CCNC(CC)=O)C)cc(C)cc2c1NCCC2C 18426,N1(C(CC2(C)CN(C(c3ccc4n[nH]cc4c3)=O)C2)=O)CCCCC(C)(F)C1 18427,N1(C(CCCC2C(C)C2)=O)CC(CNC(=O)C2=CSCCO2)OC2(CCC2)C1 18428,c1(CC)c(OC(C)C)cccc1C(N1CC(CNC(=O)CC2CCCCO2)C1)=O 18429,C1(C(N2CC(CC)C2)=O)(CNC(=O)COc2ccsn2)CC12CCC2 18430,N#Cc1cnc(C(=O)NCC2C=CC(NC(=O)CC3(O)CCCCC3)C2)c(Cl)c1 18431,CC(O)C(C)C(=O)N1CCN(C(=O)C(CN(C)C)N(c2ccccc2)C)CC1 18432,C(c1cncc(OC)c1)=CC(=O)NCC1C(NC(C2CC(C)(CC)C2)=O)CC1 18433,N1(C(CC(C)C(F)(F)F)=O)C(C)CC2CN(C(=O)Cc3c(Cl)cnn3C)CC12 18434,n1(CC)cnc2c(N3CCC(CCNC(c4ccn(CC#N)n4)=O)C3)ncnc12 18435,c1(C(N2CC(C)C(NC(=O)C=CC3(C)CCOCC3)C2)=O)cc2cnn(C)c2s1 18436,C(C(C)(CC)N1CCOCC1)NC(=O)NCCC(OCC)OCC 18437,c1(C(N2C(CCNC(C3CC4C=CC3O4)=O)COCC2)=O)cc(Cl)ccc1Cl 18438,c1(C(N2CC(OCC(=O)OCC)C(c3nccn3C)C2)=O)cc2occc2s1 18439,C12(C(N3CC(CNC(c4c(CC)occ4)=O)N(C)CC3)=O)CCCN(CCC1)C2 18440,c1(C(=O)NC2CCC(NC(C(CC)(C)C#N)=O)C2)cnn2c(Br)cccc12 18441,C1(CC)C(C)CCN1C(c1cccc(OCCOC(=O)N(C)C)c1)=O 18442,c1(-c2c(C)cccc2)nc(=NC(C)(C)CCNC(=O)CC2CCC3CC3C2)s[nH]1 18443,c1(N2CC(CNC(C(CCC)NC(N)=O)=O)OCC2)ncc2c(ncn2C)n1 18444,C(C1=NOC2CC12)(c1nnnn1C1CC(F)(F)C1)NCC(C(C)C)(C)C 18445,C(=O)(CCCCCCSC)N1C(CNC(C(C=C)(C)CC)=O)CC2CC21 18446,c1(C(N)=O)cccc(C(=O)NC2CC(NC(C3(Br)CC3(F)F)=O)C2)n1 18447,C(c1nc2ccccc2s1)=CC(N1C2(CNC(CC(CCC)O)=O)CC(C1)C2)=O 18448,CCC(CCCC(=O)NC(C)CCO)NC(=O)Cn1cc(C#N)cn1 18449,c1(CC(=O)NC2CC(F)(CNC(=O)Cc3ccccc3O)C2)cc(F)ccc1Cl 18450,N(C1CCc2cc(Br)ccc21)CC(c1c(OC)ccc(C)c1)=O 18451,N12CCCN(C(C)C1)C2=O.c1(OC(CCC#C)=O)nc(C)c(C(C)(C)C)s1 18452,c1(CN(C(CC2N(C(C3CN(CC)C3)=O)CC2)=O)CC)cnccc1C 18453,c1(C(=O)NCC2CCN(c3ccnc(C(CC)C)n3)C2)nc(C)ccc1C 18454,N1(C(C(C)OCC2CC2)=O)CCCC(C)(CNC(c2ncccc2F)=O)C1 18455,Cc1coc(C=CC(=O)NCC(CC(C)C)NC(c2coc(Br)c2)=O)n1 18456,C(c1ccccc1Cl)=C(C)C(=O)NC1CCN(C(=O)CC2CCC(C)C2)CC1C 18457,Cc1nccn1CCC(=O)NCC1CC(NC(c2ncoc2C(C)(C)C)=O)C1 18458,c1(NC(C(CC)N(C)C(C2CC2[N+](=O)[O-])=O)=O)cc(C)cc(O)c1 18459,CON1CC(C(=O)NCC2(C(N3CCC(OCC(N)=O)C3)=O)CC2)CC1=O 18460,C1(NC(C2C(CC(C)C)C2)=O)CCCC(CC(=O)NCCc2cc(O)ncn2)C1 18461,C(=O)(C(COC1(CO)CC1)C(F)(F)F)N1CCC(NC(C(C)OCC#C)=O)C1 18462,Cc1cc(=NCCN2CCC(C)CC2)[nH]c(NC2CCCC(F)C2)n1 18463,CCC(C)CC(C)C(=O)NCCCOCCN(C(=O)CSc1ccc(C)nc1)C 18464,C(=O)(CCCC(O)c1ccccc1)NCCC(C)NC(C1CCC(N=[N+]=[N-])C1)=O 18465,N1(C(C2C(C)(CC)C2)=O)CCCCC12CC(NC(=O)Cn1ccnc1C)C2 18466,N1(C(c2c(=O)ccn(C)c2)=O)CCN(C(C2(F)CC2(Cl)Cl)=O)CC12CC2 18467,C1(NC(c2c(C)nn(C)c2)=O)CCCCC12CCN(C(=O)COC1CCOC1)C2 18468,C1(C(=O)NC2C(C#C)CCC2)CNC(=O)CN1C(=O)COC1CCC1 18469,Cc1ccc(C(N2CC(C)CC(O)C2)=O)cc1S(=O)(=O)NCCC(=O)O 18470,N(C1CCCc2c(F)cccc21)C(C(=O)NCCCC=C)=O 18471,C#CC1CN(C(C2CN(C(c3nscc3C)=O)CC2(C)C)=O)CCN1C 18472,C1(CC)CC(C(=O)NC2(CNC(c3ccc(Cl)nc3C)=O)CC2)CCC1=O 18473,c1(C(N2CCC(Cc3ccccc3Cl)CC2)C(=O)NCCC#N)nc(Cl)sc1Cl 18474,C1(NC(C=C2CCC(C)CC2)=O)CCN(C(c2cc(Cl)n(C)n2)=O)C12CC2 18475,c1(C(N(C)CCN(C)C(C2CC(C(F)(F)F)C2)=O)=O)ccoc1I 18476,N1(C(C(C(C)(C)C)=O)=O)CC(CNC(C2CC(F)(CO)C2)=O)CC12CCC2 18477,N1(C(CC2C(C)(C)C2)=O)C2CCC1CN(C(c1cc(C3CC3)ccn1)=O)C2 18478,c1(CC)nccc(=NCCOCCN(C(=O)CCc2cc(C)cc(C)c2)CC)[nH]1 18479,CC(C)C(C(=O)NCC1CN(C(c2ccc(Cl)cn2)=O)CCO1)c1cnn(C)c1 18480,N1(C(C(C)=C2CC2)=O)CCC2(C1)CN(C(c1ccc(F)c(O)c1F)=O)C2 18481,C1(C(=O)NCC2(NC(c3cncc(C)n3)=O)CC2)CCC2C1C2(F)F 18482,n1(CC)nc(CN2CC3CC2(C)C3)c2c1CCOC2 18483,C1(NC(C2(CCOC)CC2)=O)CN(C(c2cncn(C)c2=O)=O)C2CCCCC12 18484,C#CC(C)(C)C(=O)NC1CCC(C(=O)NCCC2CC2C)CC1 18485,Cc1nn(C)cc1CCC(=O)NCCC(C)NC(c1[nH]ncc1C#N)=O 18486,c1(CN(C(=O)C(=O)NC2CCCCC2n2cccn2)CC)ccc2c(c1)COC2 18487,c1(C(=O)NC(CN(C(COCCCC#C)=O)CC)C)ccc2c(n1)NC(=O)CO2 18488,C1(C)(C(=O)NCCOCCCNC(C(C2CCOC2)OC)=O)CC2(CCC2)C1 18489,C(=O)(C1=CC2CCC1C2)N(CCN(C(c1cnn(-c2ccccn2)c1C)=O)CC)CC 18490,C1(CNC(C(C)(C)SC(F)(F)F)=O)CN(C(c2cnns2)=O)CCO1 18491,C1(OC(C)C(=O)NC(=O)Nc2ccccc2)CCC(c2nccn2C)C1 18492,N1(c2nnc(CC)s2)CCC(NC(=O)CNC(c2cscn2)=O)C(C)C1 18493,N1(C(c2c(CC(C)C)onc2)=O)CC(NC(C2COC(C)C2)=O)C2CCCC12 18494,N1(C(CNS(CC)(=O)=O)=O)CC(CNC(c2cc(F)c[nH]2)=O)C(O)C1 18495,c1(COC(C2(c3ccc(OC)cc3)CCOCC2)=O)cnc(F)cc1C 18496,C(CCN=C(NCc1cncc(O)c1)NC1CCOC(C)C1)OC(C)C 18497,C1(CN(C)C(C2C(C)(C)C2(F)F)=O)CN(C(c2nnn(C)n2)=O)CCO1 18498,C#Cc1ccc(C(N2CCCC2CN(C(=O)C(F)CC)CC)=O)c(OC)c1 18499,C(=O)(CCC(F)(F)CN=[N+]=[N-])NCCC1N(c2nnc(CCC)s2)CCC1 18500,N1(C(C=CCOC(C)(C)C)=O)CCCC2CCN(C(=O)C3=C(Cl)CCC3)CC12 18501,Cc1cnc(C)c(C(=O)NCC2CC2CNC(c2n[nH]cc2C(C)C)=O)c1 18502,c1(C(=O)NC2CC(C)N(C(=O)CCC(C)(C)O)C2)ccc(C#N)c(Cl)c1 18503,C1(C(=O)NCC(CC(C)C)NC(c2[nH]cc(CC)c2)=O)CC2(C1)CC(C#N)C2 18504,c1(CC(=O)N(c2ccc(Cl)cn2)C2COC2)ccc(C2CCNCC2)cc1 18505,c1(OC)cccc(C(N2CCC(N(C)C(C3C(C)(C)C3(F)F)=O)C2)=O)c1[N+](=O)[O-] 18506,C(=O)(N(OC)C(C)C=O)C1CC(N(C(=O)C2=NN(C)C(=O)CC2)C)C1 18507,N1(C(c2cc(COC)sc2)=O)CC(CNC(c2cscc2COC)=O)C(C)C1 18508,C(C1CCCCCC1)=CC(=O)NC1(CCNC(C2(C)CCCOC2)=O)CCCC1 18509,C1(C(C)(C)C)CCN(C(=O)C(=O)NCC2CCCC2)C(C(=O)O)C1 18510,c1(NCC(COC)(F)F)[nH]c(=NCCC2CCOC2)nc2c1ncn2C(C)C 18511,N1(C2(c3nc(C)oc3)CC2)CCN(c2ccc(C)c(C)c2)CC1C.c1nnnn1C 18512,C(=O)(C(C)C1=CCCC1)NC(CCCNC(C=CC=CC)=O)c1ccccc1 18513,C1(CNC(CCCOC)=O)CCC(F)(CNC(=O)CC2CCCC(C#N)C2)CC1 18514,c1(C(C)=O)cc(C(=O)NCCCC(C)NC(C23CCC(OC)C2C3)=O)n(C)c1 18515,N1(C(C(CCCC)C)=O)Cc2n[nH]cc2C1C(=O)NCCc1nnc(C)s1 18516,CN1CCC(C)(C(=O)NCC(O)CCNC(=O)C(CN(C)C)N(C)C)CC1 18517,c1(CN2CC(NC(=O)CCN3CCCC3)CC(F)(F)C2)ccc2c(c1)OCCO2 18518,N1(C(C2C(CCC)C2)=O)CCOC2CN(C(c3ccc(CF)cc3)=O)CC12 18519,N1(C(C2(CC#C)CC2)=O)CCc2nc(O)cc(C(=O)NC3CCN(C)C3C)c2C1 18520,C12(C(=O)NC(C)CCNC(C3C4(CC4)C34CC4)=O)CCCC1OCC2 18521,c1(COC(C23CCC(OC)C2C3)=O)ccc(F)cc1C#N 18522,c1(OCC)cccc(C=CC(=O)NC2CCCN(C(C3(C)CNC(=O)C3)=O)C2)c1 18523,CC1(C)CCN(C(=O)C=Cc2cccnc2)CC1CNC(=O)Cc1cc(Cl)cs1 18524,CC1CCCN(C(=O)CC(F)(F)c2ccccc2)C1CNC(=O)CC1OCCO1 18525,S(=O)(=O)(c1c[nH]ccc1=NCC1CCC(C)(C)O1)NCc1c(Cl)cn(C)n1 18526,N1(C(CNC(CC)=O)=O)Cc2nccn2CC(NC(=O)CC2CCCCO2)C1 18527,c1(OCCC(=O)NC2CC2NC(=O)C(C2CCCCCC2)O)ccc(F)cc1F 18528,C1(C(N2CCC(c3ccon3)C2)=O)COC2(C1)CN(C(c1cccnc1O)=O)C2 18529,C#Cc1ccnc(C(=O)N(CCCOCCNC(=O)C(C(C)CC)OC(C)=O)C)c1 18530,C(CC(=O)N1CCN(C)CC1C)(C(C)OCC)NC(CCOCCC)=O 18531,C1(NC(c2cc[nH]n2)=O)CN(C(c2cscn2)=O)C2(CCC2)C1 18532,C1(C(=O)NCC2OCCN(C(C3(n4cccn4)CC3)=O)C2)CCCCNC1=O 18533,c1(C(=O)OC)cc(CN2CCOC(c3nc(C(F)(F)F)n[nH]3)C2)cc(N)c1 18534,C(=O)(N=c1[nH]nc(Cl)c(C)c1C)c1c(C)nc(-c2ccccc2)s1 18535,N1(C(C2C(NC(C(C)NC(CC)=O)=O)CC=CC2)=O)CCOC(C)C1C 18536,C1(C(=O)NC(C)C=CC(=O)NCCN2CCC2)OCCCC1(C)C 18537,S(=O)(=O)(c1ccc(S(=O)(=O)N(C)C)cc1)NC(C)(C)C(=O)CC#N.N 18538,C=Cc1ccc(CNC2CCC23CNC3)cc1 18539,c1(C(=O)NC2CN(C(Cc3ccc(C)o3)=O)CC2(C)C)cc(Cl)cc2c1CCC2 18540,Cc1cc2c(cc(C(N3CC4CCN(C(=O)CO)C4C3)=O)n2CC2CC2)s1 18541,C1(NC(c2c(C#C)cn(C)n2)=O)CCN(C(=O)C(C)OCCOCC)CC1(C)C 18542,C12(NC(C3CN(C(CS(C)(=O)=O)=O)CC34CC4)=O)CCC(C1)C(O)C2O 18543,c1(C(N2CCC(NC(c3ccn4c3CCCC4)=O)C2)=O)cc2c(cc1Cl)NCC2 18544,C=CCC(CC=C)C(=O)N1CCCC1C1(NC(=O)C=Cc2cncnc2O)CC1 18545,C1(O)(CNC(Cc2c(C)cccc2)=O)CCCN(C(c2c(C)noc2C)=O)CC1 18546,c1(SC)cc(C(N2CCC2CNC(=O)C2CC2)=O)nn1C 18547,C(=O)(C(F)CCC(C)(C)C)NC(C(C)C)CCNC(c1noc2c1COCC2)=O 18548,C1(C(N2C(C)(CC(=O)NC3(CO)CCOCC3)CC2)=O)(CC)CCOCC1 18549,C1(C(N2CCOCC2)=O)CN(Cc2ccnc(Br)c2)CC(F)(F)C1 18550,c1(CC(=O)N(C(C)CCNC(c2c[nH]c(Br)c2)=O)C)cccc2ncccc12 18551,Cc1cccc(CNC(C2CCN(c3cccc(C(N)=O)n3)CC2)=O)c1N 18552,Cc1ncn(C)c1C(N1CC(n2cc(CNC(c3csc(=N)[nH]3)=O)nn2)C1)=O 18553,c1(C(=O)NC2C(CNC(C3C(C)(C)C3C(F)F)=O)CCCC2)cc2occc2[nH]1 18554,C1(NC(Cc2c(C)cco2)=O)CCCCCN(C(c2ccc3cnnn3c2)=O)C1 18555,N1(C(C=C(C)C(C)(C)C)=O)CCCCCCC1C(N1CC2CCOC2C1)=O 18556,CC(C(=O)NC1CCN(C(=O)C(c2cc(F)ccc2F)=O)C1)C1=CCCC1 18557,Cc1oc([N+](=O)[O-])cc1C(N1CCC(O)C(NC(=O)C=CCO)C1)=O 18558,N1(C(c2[nH]n(C)c(=O)n2)=O)CCC(NC(c2ccc3ccsc3c2)=O)C(C)(C)C1 18559,N1(c2nnc(C(C)C)o2)CCC2(CC1)CN(C(=O)C(F)C1CCOC1)CC(C)O2 18560,c1(N2CCN(C(C)C)CC2)ncc([N+](=O)[O-])cc1F.c1(C2C(C)N2)ccc(F)cc1 18561,N1(C(C2=CC(C)(CC)C2)=O)CC2CCCC2(NC(c2ccn(C)c2)=O)C1 18562,N1(C(C2CC(C)SCC2)=O)CCC2(C1)CN(C(=O)Cn1cccc1)CCO2 18563,n1(CC)cc(C(N2CC(C(O)C(=O)NC3CC(C(C)C)C3)C2)=O)nn1 18564,C1(NC(c2ccc(C)nn2)=O)CN(C(C2CC2C(C)O)=O)CCC12CCC2 18565,N1(C(C(C(C)C)n2cnnn2)=O)CC2(CCC2CNC(=O)C(=O)N(C)C)C1 18566,N1(C(C2=CCCN(CC)C2)=O)CCSC2(CCOCC2)C1 18567,c1(C(=O)NCCCCNC(C(C)OCOC)=O)cnn(CCCN2CCCC2)c1 18568,C1(NC(c2ccc(C)o2)=O)CCCCC12CCN(C(c1cncc(F)n1)=O)C2 18569,C1(CC(N2CC(CC(C)NC(CCNS(CC)(=O)=O)=O)C2)=O)CCCN1C 18570,N#Cc1ccc(C(N2CC3CC3(NC(=O)CCC3CCCCCC3)C2)=O)[nH]1 18571,c1(CC(=O)NC2C(COCC(=O)NC3CC(F)(F)C3)CC2)ccc(C(F)F)cc1 18572,c1(C(N(CCN(C(C(CC)C)=O)C)C)=O)cccnc1-n1ccnn1 18573,c1(-n2cc(C3(F)CCN(C(CC=CC)=O)C3)nn2)ccc2c(c1)OCCO2 18574,CONC(=O)C(=O)N1CCC(O)(C(C)NC(=O)C(N2CCCCC2)C)C1 18575,c1(C(=O)NCCC(C)CCNC(=O)CS(C)(=O)=O)cc(C(F)F)cc(F)c1 18576,C1(NC(CCC(C)OC)=O)C(C)CCN(C(=O)COCCN(C)C)C1C 18577,C1(C(N(C)C)=O)CCCC(C(N2CCN(C(c3cccnc3CO)=O)CC2)=O)C1 18578,C(=O)(C1=CCS(=O)(=O)C1)N1CCC(O)(C(C)CNC(c2cc(O)nc(Cl)c2)=O)C1 18579,CS(=O)C=CC(=O)N1CCC(CCCNC(=O)C(C)(F)c2ccon2)CC1 18580,c1(C(=O)NCC2CC(NC(=O)Cn3ccnn3)C(O)C2)coc2ccc(F)cc12 18581,C(CS(=O)(=O)c1cccs1)NC(=NCCCOCCOC)NC1CCCCC1C 18582,N1(C(C(C)OCOC)=O)CCC2(CCC(NC(c3ccc4n[nH]cc4c3)=O)C2)C1 18583,C1(Cn2c(N3CCC(C#C)(O)CC3)nnn2)CC2(CO1)CC(F)(F)C2 18584,c1(CC)cc(C)c(C(N2CCN(c3cccs3)CC2)C(=O)NCCOC)cn1 18585,c1(CNC(CCN2CCC(CCNC(c3ccc(C)s3)=O)C2)=O)cn(C)nc1C 18586,c1(SCC)ncc(C(=O)NCCCC2C=NNC2=O)o1.C1CC(=O)NCCCO1 18587,CC1CC(C(=O)NC2CCCC2CN(C)C)N1C(C1CSC1)=O 18588,c1(C(=O)NCC(C(N2CC(C)(CC)C2)=O)C)n[nH]c2c1COC2 18589,C1(Nc2cccc(NC(NNC(=O)C3C(C)CCO3)=O)c2)CCn2ccnc2C1 18590,N1(CC(CNc2cccc(C)n2)O)CCN(C2CC2)CC1C 18591,c1(C(=O)NCCN(C(C2CC(CCC)C2)=O)C)occ(C)c1C 18592,N1(C(CC2(NC(C)=O)CC2)=O)CC(O)(C(F)C(=O)NCC2(OC)CC(C)C2)C1 18593,N1(C(C(CNC(C(CC2CC2)OC)=O)C)=O)CCc2ccc(C#N)cc21 18594,c1(C(=O)NCC2CCN(C(C3(CCCC)CC3)=O)CC2O)cccc2c1CCN2 18595,c1(C(N2CCC(C)(C(=O)NC(C(C)SC)C)C2)=O)cnc2cc[nH]c2c1 18596,c1(CC(=O)NC2C(NC(C3(C#N)CCCC3)=O)COCC2)ccc2c(c1)CCO2 18597,N1(C(c2c(C)cc(C)s2)=O)CCC(CNC(c2c[nH]nc2C2CC2)=O)C(C)C1 18598,C(c1ccc(Cl)c([N+](=O)[O-])c1)=CC(=O)NCC1N(C(c2nc(C)sc2)=O)CC1 18599,N1(C(CCSCCCC)=O)CC(NC(C2CCCN2C)=O)CC1(CC)CC 18600,C1(C(=O)NCc2snc(C)n2)CN(C(C2CNC(=O)N2)=O)CC1C(C)C 18601,C(N=c1[nH]c2c(c(=NC3CC4(CC4)C3)[nH]1)CSC2)C1(C)CC1(F)Cl 18602,N1(C(=O)NCc2cncn2-c2cccc(Br)c2)CCCN(CCO)CC1 18603,c1(COC)nn(C)cc1C(N1CCCC1(C)CNC(c1c(CO)n[nH]c1C)=O)=O 18604,N1(CC(N2CCN(c3ccc(C)cc3Cl)CC2)=O)CCN(C(C)C)C(C)(C)C1 18605,N1(C(CNC(=O)Cc2cnns2)=O)CCN(C(=O)CC2CCC(=O)NC2)CC1 18606,c1(-c2n(-c3cccc(C)c3)nc(C)n2)ccnc(P(C)(C)=O)c1 18607,C1(NC(c2cc(OC)no2)=O)CC2CCC1CC2NC(C1CCCC1(C)C)=O 18608,C=C(C)C(C)(O)C(=O)N1CCCC(C)(NC(c2cnc(S)n2C)=O)C1 18609,Cc1ccc(Br)c(N)c1C(N1CC(N2CCCCCC2)C1)=O 18610,CCC(C)C(C(=O)NCC1CC2(CC2)CO1)NC(=O)Cn1cnnc1O 18611,N1(C(CN(CCOC)C)=O)C2CCC1CC(NC(C1(C)CCC(O)CC1)=O)C2 18612,N1(C(C(C)Cc2ccco2)=O)CCCC2(CCCN2C(c2csc(=N)[nH]2)=O)CC1 18613,CC1(CNC(=O)COC2CC(NC(=O)CC3CCCC(=O)C3)C2)CC2(CCC2)C1 18614,c1(C(=O)NCC(CC=C)NC(C2COCCN2CC)=O)ccc2nccnc2n1 18615,C1(C(=O)NC(C)CCCNC(c2cc(C(C)(C)C)ccn2)=O)COC2(CCC2)C1 18616,CC1CCC(Cl)=C(C(=O)N2CC(NC(=O)C(C)(F)F)C(C)C2)C1 18617,c1(CC)ccc(C)cc1C(N1CCCC1C(C)NC(c1[nH]nnc1C)=O)=O 18618,C1(C(=O)NCC2(C(=O)NCCN(C)CCO)CC(C)(C)C2)CC(=O)NC(=O)C1 18619,C1(NC(=O)C(O)C(F)F)CN(C(=O)Cc2ccc3nonc3c2)C2(CCC2)C1 18620,C1(N(C(c2cccn2C(C)C)=O)CC)CCCN(C(c2ccc(CF)cc2)=O)C1 18621,c1(C(=O)NC2C(NC(c3ccc(C4OCCO4)cc3)=O)COC2)ncc(F)cn1 18622,Cc1cc(C(=O)NCCNC(c2cnc(C3CC3)s2)=O)c(C)n1CC(F)(F)F 18623,c1(C(N2CC(C(=O)NCc3nn[nH]c3C(F)(F)F)C2)C)ccccc1F 18624,C1(C(CSC)NCc2ccc(C)cc2C)CCC(F)(F)CC1 18625,c1(CN(CC(=O)Nc2cc(C(=O)OCC)n(C)n2)CCOC)cc(F)ccc1F 18626,C1(F)(C(=O)NCCC2(CNC(C3CC=CCC3)=O)CC2)CC1(Cl)Cl 18627,C(=O)(C1CCCc2ncnn21)N1CCC(CC(=O)Nc2cnc(C)c(F)c2)C1 18628,C(=O)(CC(C)O)NC(CNC(C(C)OCCCC)=O)(C)C1CCC1 18629,c1(C(=O)NC(CC)CNC(c2ccc(C(C)C)cc2C)=O)c(C)nc(C)nc1C 18630,Cc1nccc(C(=O)NCC2(CNC(c3cscc3F)=O)CCCCC2)c1N 18631,c1(C(=O)NC2C(NC(C(C)C#N)=O)C2)c(F)ccc(F)c1Cl 18632,c1(CCNC(=O)CCC2CCCN2C(=O)CC2CCC3CC23)cccnc1F 18633,N1(C(CC(C=C)(C)C)=O)CC2CN(c3ncc(C(=O)OC)cc3Cl)CC2C1 18634,c1(C(=O)NCCN(C(=O)Cc2ccon2)C(C)C)cc(Cl)n(C)n1 18635,N1(C(c2c(OC)csc2)=O)CCOCC1C(=O)Nc1cncc(C(F)(F)F)c1 18636,C1(CC(N2C(CNC(C(C)n3cccc3)=O)CCC2)=O)SC(=N)NC1=O 18637,C(CCC(C(=O)NCc1cccc(Br)c1)N1CCCC1CC(C)(C)[N+](=O)[O-])OC 18638,C1(N(C(=O)CCCn2cccn2)C)CCCN(CCCN2CCCC2=O)C1 18639,c1(C(=O)NC(CC(=O)NC2CC(OCC)C2)C2CC2)cc(OC)n(C)n1 18640,C(CC(F)(F)F)CC(=O)NCc1cn(C2CCN(C(=O)CC3CC(F)C3)C2)nn1 18641,c1(C(=O)NCC23CC(NC(C(c4ccccc4)OCC)=O)(C2)C3)cnn(C)c1F 18642,C1(NC(c2cccn(C)c2=O)=O)CCCC12CCN(c1ncnc(=N)[nH]1)CC2 18643,C1(n2cc(CC=CC)nn2)CCCCC1NCc1cnn(CCO)c1N 18644,C1(CNC(c2cc(C)[nH]n2)=O)CC2CC2N1C(=O)CC(F)(F)Cl 18645,C(CC(=O)NCc1c(C)cccc1O)(C(F)(F)F)NC(C=CC=CC)=O 18646,N1(C(c2c(CC)nns2)=O)CC2CCCC(C1)N2C(=O)C(C)(O)COC 18647,c1(N(C(=O)C(n2cc(-c3nccs3)nn2)C)CC)nc(O)c2cnn(C)c2n1 18648,C(=O)(C(C(C)C)NC(=O)COCCSC)NC(CC)CO 18649,C1(C(=O)NC2C(NC(C(C)=CC)=O)COC2)CCCN(C(N2CCCC2)=O)C1 18650,NS(=O)(=O)c1sccc1C(=O)N(CCNC(C1COCCO1)=O)C1CC1 18651,c1(C(=O)NCCCC(CCC)NC(=O)CNS(N)(=O)=O)cc(F)cc2nc[nH]c12 18652,C1(CCNC(c2c(CC)ocn2)=O)CSCCN1C(C1CCCC1C)=O 18653,c1(C(=O)NCC2OCCN(C(C(C(C)OC)O)=O)C2)ccc2c(n1)NCCO2 18654,c1(C(c2n(CCC)nnn2)NC(C(N)=O)C2CC2)ccc(C(F)F)cc1 18655,C12=CC(=NCC3CCCN3C1=O)NC=N2.C1(C(=O)OC)CC1C 18656,c1(CC(=O)NC(C(=O)NCCC(C=C)C)(C)C2CCC2)ccccc1C 18657,N1(C(C(=O)NCCOC)=O)CCOC2CCN(C(=O)C(C)CC3CC3)CC12 18658,C1(CN(C(C(C=CCCC)O)=O)C)CN(C(=O)C=CCCCCC)CCO1 18659,c1(C(=O)NC2CCN(C(c3cn(CCC)nc3)=O)C(C)C2)ccc(C)c(C)c1N 18660,CC1CCC(CNC(c2cc(CNC(C3(c4ccno4)CC3)=O)cs2)=O)N1C 18661,C1(CN(C(C(C)(C)OCC)=O)C)CCC(CNC(=O)CC(O)C2CCCC2)CC1 18662,c1(CNC(CCN(C(=O)Cc2ccc[nH]2)CC#C)=O)cc(C)cnc1O 18663,N1(C(C=C(C)CNC(=O)CCn2ccc(C)n2)=O)CCCCC1C1CCC1 18664,N1(C(c2cc(OC)nn2C)=O)CC(C)N(C(c2cc(C)n(C)c2)=O)CC1C 18665,Cn1c(C(=O)NCC2CC(NC(=O)CSCc3ccccn3)C2)cnc1Cl 18666,N1(C(c2c(N3CCCCC3)cccc2Cl)=O)CC2CCC(C1)C2.N1CCCC1 18667,c1(C(N(CC(C)(C)O)CCOC)=O)cc(C(F)F)ncc1F 18668,C1(OCC)CC(NC(=O)C(N2CCCC2(CC(C)C)CC(C)C)=O)C12CCC2 18669,c1(NC(C2(F)CN(C(c3cc(Br)ccc3Cl)=O)C2)=O)cnc2ccc(F)cn12 18670,c1(CNC(c2n(CC=C)nnn2)c2ccn(C3CC3)n2)cccc(Br)c1.OC(F)F 18671,N1(C(CSCCNC(c2cccn(C)c2=O)=O)=O)CC2(CC=CC2)C1 18672,N1(CC(=O)NCCOCC(=O)NC2CC2(F)Cl)CCCCS1(=O)=O 18673,N1(C(c2scnc2C2CC2)=O)CC2CCC(C1)N2C(C1CCCC1O)=O 18674,C(=O)(C(F)(CNC(=O)CCc1nncs1)C(C)C)NCCC(=C)C 18675,C1(CN(C(c2cc(Cl)cn2C)=O)CC)CCN(C(c2nncs2)=O)CC1 18676,C1(NC(C2(C#C)CCC2)=O)CCN(C(c2cc(CC)c[nH]2)=O)CC1F 18677,C(=O)(CCCC(=O)N1CCCN(C(=O)CNC(=O)CCCCO)CC1)OC 18678,c1(C(=O)NCC2CC2)cc2c(s1)CCN(C(=O)CN1CCCCC1=O)C2 18679,CC(O)C(C)(C)C(=O)NCC#CCNC(C1CC(O)CN1C(=O)OC(C)(C)C)=O 18680,C1(Cc2c(F)ccc(OC)c2)CCN(C(=O)CC(C)c2ccccc2)CCC1CSC 18681,N1(C(C(C)O)=O)CC(C(=O)Nc2ccc(OCc3ccccc3)nc2)CC(C)C1 18682,C1(C(=O)NCC2CN(C(=O)CO)CCC2(F)F)Cc2cncn2C(=O)N1 18683,c1(OC)cccc(NC(C2(C)CCN2C(c2cccnc2O)=O)=O)c1 18684,C1(C(=O)NCCNC(c2cc(Cl)sc2Cl)=O)COC2(CO)CC1C2 18685,C1(NC(C2CN(S(CC)(=O)=O)C2)=O)CC(F)CN(C(c2csc(C(F)F)n2)=O)C1 18686,C1(NC(C2CC23CC3)=O)C2COCC1CN(C(=O)CCc1ncc(F)cn1)C2 18687,Cc1ccc(Cl)c(C(=O)NCCCN(C(=O)CN2CCC2C)C2CC2)c1 18688,C1(CN(C(=O)CC2(C)CC2(F)Cl)C)CCN(C(C2(O)CCCCC2)=O)CC1 18689,c1(OC)ccc(N)c(C(N2CCC(NC(C3CC3(C)C)=O)C2(C)C)=O)c1 18690,c1(C(=O)OC2CCS(=O)(=O)CC2)cc(Br)cc2c1CCN2 18691,c1(C(=O)NCC(C)(C)NC(c2cnn[nH]2)=O)ccc(F)c(Cl)c1N 18692,CN1CC(NC(=O)CNC(=O)CNC(c2n[nH]c3c2CCC3)=O)C2(CC2)C1=O 18693,CC1(C)OCCCC1C(=O)NCC1CN(Cc2ccccc2)CCCO1 18694,N1(C(CSC)=O)CC(NC(=O)Cn2nc(C)c3cccnc23)C2CCCCC12 18695,c1(C(C(=O)N(C2CN(C(=O)CC3CCCC(O)C3)C2)C)(C)C)cccc(C#N)c1 18696,C1(NC(C(C(C)(C)O)F)=O)CC(C2CCN(C(=O)CCc3nc(=N)[nH][nH]3)CC2)C1 18697,C12(CC(=O)N(C3CCCC3)CCCNC(C(C)O)=O)CC3CC(C1)CC(O)(C3)C2 18698,c1(NC2CCC2)ccc(C(=O)NC2C(NC(C(C3CC3)OCC)=O)CC2)nc1 18699,CN1CC(C)(C(N2CC(N(C)C(c3cc(C4CC4)ns3)=O)C3(CC3)C2)=O)CC1=O 18700,C(=O)(C(CC(C)(C)C)NC(c1ccc(NC)cc1)=O)NC(C(=O)NC)(C)C 18701,C(C(C)C(=O)NC(C)CNC(c1cnc(-c2ccoc2)s1)=O)OC 18702,c1(CC)cccc(C)c1C(N1CCCC(O)(CNC(=O)CC2CC2C2CC2)C1)=O 18703,CC(CC(=O)NCC1CC1CC(=O)NCC1(SC)CC=CC1)C1CC1 18704,C1(NC(c2cn(CC3CC3)nn2)=O)CCCN(C(c2ccc(Cl)nc2)=O)CC1 18705,Cc1cc(C#N)nc(N2CCC(CNC(=O)CCc3ccc(O)nc3)C(C)C2)n1 18706,c1(C(=O)NCC(c2ccccc2Cl)N(CC)CC)ccc2c(c1)CC(=O)N2 18707,c1(CC)cc(C(=O)NCC2CCN2C(C2(F)CCCN(C)C2)=O)cn(C)c1=O 18708,c1(CNC(c2ccc(C)c(F)c2)=O)c(O)cc(O)cc1O 18709,Cc1cc(-c2ccnc(NC(c3ccccc3N(C)C(C)C)=O)c2)ccc1F 18710,N1(C(Cc2c(C)cccc2)=O)C2CCCC1CN(C(C1CCN(C)C1)=O)C2 18711,n1(CC)cc(Cl)cc1C(N1CC(CCNC(c2ccc(C#N)[nH]2)=O)C1)=O 18712,N1(C(C2(CC)CCC2)=O)CC2(CCN(Cc3nnc(C(C)C)s3)C2)C1 18713,C1(C(=O)NCCCc2c(C)n[nH]c2)CCN(C(c2[nH]nnc2C(F)F)=O)CC1O 18714,C1(C)(C(=O)NCC2(NC(C3CCCN(C)C3)=O)CC2)Cc2ccccc2C(=O)O1 18715,c1(C(=O)NCC(CC)N(C(=O)C=Cc2ccc(C)s2)C)ccc(=N)[nH]c1 18716,C1(=CC(CC)C)CCN(CCC#N)CC1.C12CCC(CC1)C(=O)N2C1CC1 18717,C(=O)(NNc1ccc(F)c(Br)c1)C(=O)OC(C)(C)C.CC1CCCCC1CN 18718,N1(CC(=O)NCCOCC)CCC(NC(C2CCOC(C)C2)=O)CC(C)(C)C1 18719,C1(NC(COCCC=C)=O)CC2(CCN(C(=O)C=Cc3cnccn3)C2)C1 18720,CCC(C)(CCNC(=O)CCCC1CCCO1)NC(=O)CC1(C)CC1 18721,c1(C(N2CC(C)(NC(C(N3C(CC)CCC3)=O)=O)C2)=O)ncccc1C 18722,c1(OCC)ccc(F)c(F)c1-c1cncc(C(N2CCC(OC)C2)=O)n1 18723,C1(CNC(C2CCS(=O)(=O)CC2)=O)CC2CCC(C1)N2C(C1CCOC1)=O 18724,C1(OC)CN(C)C(C)(C(N2CCCCC(CNC(C3(O)CCCCC3)=O)C2)=O)C1 18725,C1(CNC(c2c(C)n(C3CC3)cc2)=O)CN(C(=O)C(C)SC(F)(F)F)CCCO1 18726,N1(C(C(COC)OC)=O)CC(NC(c2ccc(OC)c(Br)c2)=O)CC1(C)C 18727,Cc1cnccc1CNC(=O)C(CCF)NC(c1cnccc1C)=O 18728,C#CCC(C)(C)C(=O)N1CCC(C)C(NC(c2cncc(C(C)C)c2)=O)C1 18729,c1(C(=O)N(C(=O)C(=O)C2CC2)C2CC2)cccc2c1OC(F)(F)O2.c12csc(n1)N2 18730,c1(OC)ccnc(C(=O)NCC(CCOC)NC(C2CC2CC(C)C)=O)c1 18731,Clc1sc(Cl)c2c1CCCC2NC1CCC2(CC1)CC(CO)C2 18732,OC1COc2c(NCc3cc(Cl)sc3Cl)cnn2C1 18733,C#CCCCCCC(=O)N1CCC(N(C(c2cc(CO)[nH]n2)=O)CC)CC1 18734,c1(C(N(CCCNC(C2CCN(CC(C)C)C2)=O)C)=O)cc(Cl)cc2c1OCC2 18735,C#Cc1cccc(CC(=O)NC2CCOC2C(N2CCNC(=O)C2CCC)=O)c1 18736,C1(CNC(C2N(C)CC(O)C2)=O)CC2(CCC2)CN1C(=O)CC1C=CCC1 18737,Cc1ccnc(C(=O)NCC2(NC(=O)C=CS(C)=O)CCC2)n1 18738,C=C(Br)CCC(=O)N1CCCCC1C(C)NC(=O)Cn1nnc(C)n1 18739,c1(C(N(CC(=O)NC2(CC(=O)OC)CC2)CC2CC2)=O)nnnn1C 18740,C=CCCCC(C)(C)C(=O)N1CCC(NC(c2ccc(C)c(Br)c2C)=O)CC1 18741,C=CCC(CC(=O)NCC(=O)N(C)C1CC1)NC(C1CCOC(CC)C1)=O 18742,N1(CC2(NC(CCOC)=O)CC2)CCN(C(C2OCCOC2C)=O)CC1 18743,c1(N(CC(CN(C)C)(C)C)C)nc(N2CCC(C)(C)C2)nc2c1cnn2C 18744,C(=O)(C(C)(C)CC(=O)OC)NCC(CC=C)C(=O)Nc1ccc(Cl)cc1 18745,n1(C(CCO)CC2(CCC#N)CC2)cnc2c(N3CC(OC(F)F)C3)ncnc12 18746,c1(C(N2C(CNC(C(C)NS(C)(=O)=O)=O)CC2)=O)ccc(C2CC2)cc1F 18747,CC#CC1CCN(C(=O)C(C)=CCNC(C2CCN2C(C)(C)C)=O)C1 18748,C#Cc1ccc(C(=O)NCC2(NC(c3ccsc3COC)=O)CCC2)cc1Cl 18749,c1(C(=O)NCCOCCNC(C(C)SCC)=O)ccc2cn(C)nc2c1 18750,C(=O)(C1CCCn2cnnc21)NC1C(CNC(c2cccc(C(C)C)c2)=O)C1 18751,CC(C)CC(C)CC(C)C(=O)C(C1(c2cn[nH]c2)CCC1)=O.N1(CCN)C(=O)CNC1=O 18752,C(=O)(N(CCC(=O)OC)OC)C1CC(NC(CC(C)OC)=O)C1 18753,c1(C(N(CCCN(C)C(C2(O)CCOC2)=O)C)=O)cccc(O)c1F 18754,Cc1ccc2oc(C(=O)NC3CC(CNC(c4cc[n+]([O-])cc4)=O)C3)cc2n1 18755,c1(-c2cccc(C)c2)cnc(=NCc2cc(C(N3CCCC3)=O)ncc2)[nH]c1 18756,C(C(CNC(=O)CCOCC(F)(F)C(F)F)C(F)(F)F)NC(c1c(CC)cns1)=O 18757,C(=O)(C#CC1(C)CCCO1)NC(C(C)NC(c1cnn(C)c1Cl)=O)(C)C 18758,CC1=NOC(C)(C(=O)NCC2(C(N)=O)CN(C(=O)CSC(F)(F)F)C2)C1 18759,C1(O)(COC)CCN(C(=O)CCOCCCNC(c2occc2C2CC2)=O)C1 18760,CCCCS(=O)(=O)CC(=O)NCC(C1CC1)NC(c1c(C)cccc1C)=O 18761,CC(C(=O)N1CCOCC1)C(=O)N1CCC1CNC(=O)CCc1cncc(F)c1 18762,N1(C(c2cc(CC)[nH]n2)=O)CCCC(CO)(NC(=O)Cn2ccc([N+](=O)[O-])n2)C1 18763,C1(CC(=O)NC2CCN(C(=O)Cc3nc[nH]n3)CC2O)CC2CCC1CC2 18764,N1(C(c2c(COC)ccs2)=O)CCCCC2(CCN(C(c3cnc[nH]3)=O)C2)C1 18765,N1(C(c2ncc(OC)cn2)=O)CCC(NC(c2cc(C)c[nH]2)=O)C(C)(C)C1 18766,c1(C(C(=O)NCC2(NC(C3C(C)(Br)C3)=O)CC2)=O)cc(F)ccc1F 18767,C1(C(C)C)CNC(=O)CN1C(C1CC12CC(NC(c1nccn1C)=O)C2)=O 18768,C1(OC)CC2(C1)CN(C(=O)C(CNC(c1ncccn1)=O)C(C)C)C2 18769,C1(NC(NCC2N(CC)CCC2)=NCCc2ccccc2)Cc2nccnc2C1 18770,C1(SC)CC(CC(=O)NCCN(C(=O)C(C)C2CCCC2)CC(C)O)C1 18771,N1(C(Cc2ncn(C)c2)=O)CC(C(=O)NC(c2nc[nH]n2)C2CC2)C2(CC2)C1 18772,O=C(C#CC1CCCC1)NCc1cc(C(=O)NCC2CC(=C3CCC3)C2)ccn1 18773,C(=O)(C1=CCC(F)(F)CC1)NC1CC2CN(C(CC(C(C)C)O)=O)C1C2 18774,Nc1cccc(C2CN(C(C3CCOC(c4ccc(F)cc4)C3)=O)C2)c1 18775,C1(NC(CCC)=O)CCC12CN(C(=O)CCC(c1ccccc1)N(C)C)C2 18776,Cc1ncc(NC(C2CN(C(c3cncc(Cl)c3)=O)CCN2)=O)c(C)c1Br 18777,N1(C(C(F)=C(C)C)=O)CCOCC(C(=O)NCc2cc(F)ccc2F)C1 18778,Nc1c(C(=O)NCCC2CCCCN2C(=O)C(O)C2CCC2)ccnc1Br 18779,CC1=CCC(C(=O)NCC2CC2NC(c2ccc(NC3CC3)nc2)=O)CC1 18780,c1(CNC(=O)COCCNC(C2C3CCCC23)=O)ccnnc1 18781,C(C(C)(C)C(=O)N1CCC(O)(CC)C1)NC(c1ncn(CC)c1)=O 18782,C1(CNC(c2cncc(CC)c2)=O)Cc2ccccc2CN1C(c1ccon1)=O 18783,Cc1cc(C#N)ccc1C(N1CCC2(CC2NC(C2CC3(CCCC3)C2)=O)C1)=O 18784,CCCCCCCCC(C)CC(=O)NCc1ccc(OC)cc1 18785,C#CC1CCCC(CNC(=O)C(C(C)C)NC(C2C(C)C2C)=O)C1 18786,C1(CC)(CNC(C2(C(F)F)CCCO2)=O)CCN(C(c2snnc2C)=O)C1 18787,C(=O)(C(C)CCCC(C)=O)NC1C2(C(N=c3ccn(C(CC)C)[nH]3)=O)C3CC1CC23 18788,N1(C(CC2(C)CN(C(c3cc(OC)n(C)n3)=O)C2)=O)CCC(O)(CF)CC1 18789,N#Cc1cc(NC(=O)NCC23CC(CCO2)C3)co1 18790,c1(OC)ncccc1C(C)NC(c1nnnn1C)C1CCC1 18791,c1(CNC(=O)NCc2cccnc2[N+](=O)[O-])cccc2cncn12 18792,N1(C(C(c2cccnc2)C)=O)CCC2CC(CNC(=O)CCF)CCC2C1 18793,C1(CC(C)C)CC(C(=O)NCCCNC(c2cc(=O)cc[nH]2)=O)CC(=O)N1 18794,C1(CC=C)(C(=O)NCc2csc(C)n2)CN(C(=O)C(C)N2CC(C)C2)C1 18795,N1(C(c2cc(OC)ncc2F)=O)C2CCCC1CC(NC(C1CC1C(F)F)=O)C2 18796,c1(C(N2C(CC(=O)Nc3c(CC)nc(OC)cc3)CCC2)=O)cc2ncccn2n1 18797,N1(C(=O)NC(Cc2cccc(C)c2)C2CC2)CCCC(O)(c2cnn[nH]2)C1 18798,C12(C(=O)NCC(CC)NC(CCN(CCCCC)C)=O)CSC(C1)C2 18799,c1(CC)nccnc1C(=O)NCC1CCN1C(=O)C(=CC1CCCC1)C 18800,C(=O)(NNc1cccc(F)c1C(=O)O)C1C(c2n(C)cc(Br)n2)C1 18801,CC1(C)CCCCC1C(=O)NCC(C)(C)CNC(c1cnn(CC2CC2)c1)=O 18802,N1(C(CCCNC(C)=O)=O)CC2(COC(CNC(=O)C(F)CC3CCC3)C2)C1 18803,S(=O)(=O)(c1ccc(N2CC(CO)C(O)C2)c(C#N)c1)NC(CCSCC)C 18804,c1(NCC(C)(C)NC(Cc2ccc(OC)cc2)=O)ccc(C#N)cc1[N+](=O)[O-] 18805,C1(NC(C(C)OC2CCCC2)=O)CC2CC1N(C(C1(O)CCOCC1)=O)C2 18806,C12(NC(CCc3ccnc(C)n3)=O)CCCC1N(C(=O)CN(C)C(C)C)CCC2 18807,Cc1cc(Cl)cc(C(=O)NCC2(NC(C3CCC(=O)N3)=O)CCCC2)c1C 18808,C=CC(CCC)CC(=O)N1CC(C(=O)NCC2CCOC(C)(C)C2)C(F)(F)C1 18809,c1(OC)cc(C)ccc1C(N1CCCC(CNC(c2cc(Cl)c[nH]2)=O)CC1)=O 18810,C1(CNC(c2cccc(CCC)c2)=O)COCCN(C(=O)CCOCC2CC2)C1 18811,c1(C(=O)NCC(O)CNC(C2CC2C2CCC2)=O)ccc2ccc(Br)cc2c1 18812,c1(C(=O)NCC(CCCC)NC(=O)C(C)CF)ccc2n[nH]c(C)c2c1 18813,N1(C(c2c(C)nc(N(C)C)s2)=O)CCC2C(CCCN2C(c2cscn2)=O)C1 18814,c1(-c2cn(CCS(C)(=O)=O)nn2)cc(C#N)ccn1.C12CCC(CC1)CC(=O)N2 18815,C1(NC(c2cc(SC)oc2C)=O)CCN(C)C12CCCN(C(=O)C=CCO)C2 18816,c1(NC(=O)OC)ccc(NC(=O)NC2CC(OC)C2(C)C)c(Cl)c1 18817,C1(C(=O)NCC2C(C)CC2)N(C(c2coc(N(C)C)n2)=O)CC12CCCC2 18818,CCC(CC(=O)N(C1CN(C(C2CC=CCO2)=O)CCC1O)C)C(C)C 18819,C(C)(N=c1[nH]c(N2CCC3(CCN(C)C3)C2)nc2ncn(C)c12)c1nc(C)sc1 18820,Cc1nnn(CC(=O)NCc2cn(CC(=O)N(CCCF)C)nn2)n1 18821,c1(CC)cc(C(=O)NC(CC)CC(=O)NCC2COCC2(C)C)ccn1 18822,C1(F)(C(N2C(CCC(=O)Nc3cnc(C)c(Br)c3)CCC2)=O)CCCCC1(F)F 18823,C1(CNC(CCSC)=O)CC2(CCN(C(c3cc(C(F)F)ccn3)=O)CC2)CO1 18824,C(=O)(CCCS(C)(=O)=O)N1CCN(C(C(C)NC(=O)NC)=O)C(C)C1 18825,c1(C(=O)NC(C2CCN(C(=O)CCc3ncc[nH]3)CC2)C)cc(Cl)cnc1O 18826,CCC(CCCC(=O)N(CC1CCC1)CC1CC1)NC(c1cc(C)cc(C)c1)=O 18827,c1(C(=O)OC)cnc(NC2CC(C)(NC(=O)C(c3ccc(F)cc3)F)C2)c(Cl)c1 18828,N1(C(CCOCC)=O)CCC(NC(C23CSC(C2)C3)=O)C1 18829,Cc1c(C(=O)NCC(C)CNC(=O)C(C(C)C)NS(C)(=O)=O)cccc1Br 18830,CCC(C)(C)C(=O)N1CCOC(CCNC(=O)CCn2cncn2)C1 18831,N1(C(c2ccc(NC)cc2)=O)CCN(C(=O)COCCO)C(CO)C1 18832,N1(C(c2c(OC)nsc2)=O)CCC(N(C)C(c2sccc2Cl)=O)CC1 18833,N1(C(c2cc(C)cc(C)n2)=O)CC(C)CN(C(C2CCCCN2C)=O)C(C)C1 18834,n1(CC)cc(C(=O)NC2C3CCN(C(c4sc(C)nc4C)=O)C23)c2ccccc12 18835,c1(CC(=O)NC2CC(C)N(C(c3cccn(O)c3=O)=O)C2)c(F)cccc1F 18836,N1(C(CCN(C(C)C)C(C2CCCC(N(C)C)C2)=O)=O)CC2CCCC(O)C2C1 18837,O=C(C1=CCCOC1)NCCCCNC(C1CCCCS1)=O 18838,CC1CCC(C)(C(=O)NCCNC(c2ccnc(Oc3ccccc3F)c2)=O)C1 18839,N1(C(C#C)C)CCN(C(=O)C(CCF)NC(c2cnncc2C)=O)CC1 18840,C(=O)(Nn1cccc1)C1C(C(=O)OC)C1 18841,c1(C(=O)NCC2C(NC(CNC(=O)OC(C)(C)C)=O)C2)cc(CCP(C)(C)=O)[nH]n1 18842,Cc1cccc(C(=O)NCCCCCCNC(=O)CC2(C)CCCO2)c1N 18843,N1(C(c2c(CNC(c3n(C=C)nnc3)=O)cco2)=O)CCC2C(CCN2C)C1 18844,N#CC1(C(=O)NCC2(CNC(C3CCCN3C=O)=O)CC2)CC2(CCC2)C1 18845,C1(C(=O)NCCC(C(C)C)NC(c2n(CCCC)ncc2)=O)CCS(=O)(=O)CC1 18846,C1(F)(CNC(c2ccnc(O)c2)=O)COCCN(C(=O)C(O)c2ccco2)C1 18847,Cc1cc(C)c(C(=O)NC(Cc2ccoc2)C(=O)NCc2ccc(C#N)s2)s1 18848,C1(C(C)C)N(C(C2CC2C)=O)CC12CCN(C(c1nc(C3CC3)cs1)=O)CC2 18849,N1(C(CC(CCC)(C)C)=O)Cc2cccc(CNC(=O)C(COC)CC)c2C1 18850,N1(C(Cc2scc(C)c2)=O)CCC(CF)(NC(=O)C(C(C)C)n2cnnn2)C1 18851,C1(C(=O)NCC2CC(F)CN2C(C2(F)CCCCC2)=O)CCCC1C1CC1 18852,c1(C(=O)OC)ccc(C=CC(=O)NC2CCN(C(=O)C=CCOC)C2C(C)C)o1 18853,C(=O)(C1=CCOCC1)NCc1c(CN2CCN(C(C(C)SC)=O)CC2)cccn1 18854,C(=O)(CC(C(F)F)C(C)(C)C)N1CCC(N(C(C(CCC2(C)CC2)O)=O)CCO)C1 18855,Cc1cc(Cl)cc(C(N2CCCC2CCNC(c2ncnn2C)=O)=O)c1N 18856,Cc1cc(N2CCSC2)ncc1S(=O)(=O)N1CCC2CCCCC12 18857,C1(C(=O)NCc2n(CC)ncn2)CC=CC(NC(=O)C(C(C)C)NC=O)C1 18858,C1(NC(CSCC)=O)CCCCC12CCN(c1nc(Cl)nc(C)c1Cl)C2 18859,c1(CCC(=O)NC2CN(C(=O)CCc3ccoc3)C2)cccc(F)c1 18860,c1(C(=O)NCCC(C)(C)NC(c2cc(OC)cc(F)c2)=O)cnc2c(c1)NCC2 18861,c1(C(=O)OC)ccc(CC(C)C)nc1N1CC2CC(NC(=O)CC3(C)CC3)C2C1 18862,c1(C(=O)NCCC2CN(C(CC3C(C)CC3)=O)C2)cc(Cl)ccn1 18863,N1(C(c2c(C(C)=O)cn(C)n2)=O)CC2CC(N(C(=O)CCCC3CC3)C)C1C2 18864,c1(OC)ccc(-c2ccnc(C(N3CCC(F)(c4cn(C(C)C)nn4)C3)=O)n2)cc1 18865,c1(C(C(=O)NCCC)N(c2cccc(OC)c2)C2CC2)sc(Br)cc1Cl 18866,c1(C(N(C(C)CNC(c2cccc(SC(F)(F)F)c2)=O)CC)=O)cc(C)n(C)c1 18867,CC1=NS(=O)(=O)NC=C1C(=O)N1CC(NC(=O)C(F)CC2CC2)CCC1C 18868,c1(C(=O)NC2CC(NC(C(C(C)C)n3ccnc3)=O)C2)nn(C)c(C(F)F)c1Cl 18869,C1(C(=O)NCC2CCN(C(c3c(CC)c[nH]n3)=O)C2)C2CCCCC12 18870,c1(NCCCC2C(O)CCC2)nccc(=NCCOC2CCOCC2)[nH]1 18871,C(=O)(CCCCCCCC1CC1)N1CC(NC(c2c[nH]c(=N)o2)=O)CC(C)C1 18872,c1(C(=O)NCC(c2cccc(C#N)c2)C)ccnc(Cl)c1N 18873,c1(NC(C2CCN(C(Cn3ncc(CC)c3)=O)CC2)=O)ccc2ccncc2c1 18874,N1(c2ncc(C(=O)OCC)s2)CCCC2(CC(NC(=O)C(C)c3ccco3)C2)C1 18875,C1(NC(c2ccc(C(C)(C)C)cn2)=O)CC2CC(NC(=O)C3=CCCS3)CC12 18876,C1(NC(CNC(CN(C)C)=O)=O)CCOC12CCN(C(=O)CC(F)(F)F)CC2 18877,C=CCCCC(=O)N(C1CCC(NC(C2(COC)C=CCC2)=O)CC1)C 18878,c1(C(N(CC(CC)NC(C(CC)C)=O)C)=O)nn2cccnc2c1Cl 18879,C(=O)(C(C)CC(F)F)NC(C(=O)NCC1(OCC)CCC1)Cc1ccoc1 18880,N1(C(C2C(OC)CCC2)=O)CCc2[nH]nc(CNC(=O)CC3(OC)CC3)c2C1 18881,C1(NC(=O)C=CC=C(Cl)Cl)CN(C(c2cnc3n2CCC3)=O)CC12CCC2 18882,Cc1csc2ncnc(N3CCC(O)C(C(=O)Nc4c[nH]nc4C#N)C3)c12 18883,C(=O)(CC(c1ccccc1)OC)NC1CC(OCC2(OC)COC2)C1.C(=O)NC 18884,C1(C(=O)NCCNC(c2cc(F)cc(N)c2F)=O)(CC)CCC(F)(F)CC1 18885,N1(C(Cc2c(C)nccc2)=O)C2CCC(C2)C1C(=O)NOC(C)C 18886,CCCC(C)CC(=O)NCCN(C(c1ccncc1CC)=O)CC 18887,c1(CNC2CC(C)(Nc3ccn4nccc4n3)C2)ccc2ncccc2n1.C1CC1 18888,CCN=c1[nH]cc(C(N2CCC(C)C(CNC(C3(C)CC3)=O)C2)=O)s1 18889,c1(C(N2CC3(C2)SCCC3NC(=O)C(F)(F)C2CC2)=O)cccc2sccc12 18890,Nc1nc2ncccc2cc1C(=O)NC1(CO)CCN(C(=O)CC2CCCC2)C1 18891,N1(CCc2ncn(C)c2)CCc2onc(C3CC3)c2C1 18892,Cc1cc(C(C)C(=O)NCC2CC3(CCOC3)C2)cc(F)c1 18893,c1(C(N2CCCOCC2C)C(=O)NCC(=C)C)cccc(C(F)(F)F)c1F 18894,N1(C(C(C2(O)CCCC2)OCC)=O)CCSC12CC(C(=O)O)C2 18895,CC1CC(NC(=O)NNC(=O)c2cn(C)nn2)CCN1C 18896,S(=O)(=O)(CCC(F)(F)F)N1CC(C)(CC(=O)NCC(=O)NC2CC2)C1 18897,N1(C(CC2C(CC)CC2)=O)CCN(CCSc2ccc(NC(C)=O)cc2)CC1 18898,c1(C(=O)NCCNC(c2c(C)nc(-c3ccc(F)cc3)s2)=O)cc(N)cnc1C 18899,C(CC(C(=O)N1CCC(NC(=O)CC2CCCC23CC3)C1)OC)OC 18900,C1(NCc2cnc(C(C)(C)C)[nH]2)CCN(c2ccccc2)C1=O 18901,C(CC(=O)N(CCCNC(=O)C(O)Cn1cncn1)C1CC1)(C(F)(F)F)OCC 18902,Cc1nsc2c1C(=O)N2.C1(C(N(CCNC2CC2)C(C)C)=O)CCCCC1C 18903,C(=O)(C1=NNC(=O)CC1)NCC1(NC(c2nccc(C)c2)=O)CCOC1 18904,N1(C(c2cncc(N)c2)=O)CCC2C(C1)CN2C(c1cccc2sccc12)=O 18905,C1(O)(C(=O)NCC2CC(NC(COC(CC)C)=O)C2)CCCC1 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19064,N1(C(c2cccc(SCC)c2)=O)CC2CCN(C(C3CCC4CC34)=O)C2C1 19065,N1(C(c2ccc(C)s2)=O)CCN(C)C(C2CC2)C1.C12CCOC1C(=O)N2 19066,C1(NC(C=Cc2nc(C)sc2)=O)CCC(O)CN(C(=O)C(C)(O)C2CCC2)C1 19067,c1(CC)cc(C(=O)NCC(C)CNC(=O)C(C(C)(C)C)n2ccnn2)ccc1Cl 19068,Cn1c(C(N2CCOC(C(=O)NC3CCC(CCO)CC3)C2)=O)ccc1C#N 19069,C1(NC(c2ccc(OCC=C)cc2)=O)CN(C(=O)Cn2cnc(=N)[nH]2)C(C)(C)C1 19070,C1(CNC(c2cccnc2C2CC2)=O)CCC(C(=O)NC2CCCC(O)C2)CC1 19071,N1(C(c2ccc(C)[nH]2)=O)CC2C3CCC(C2C1)N(c1nnc(C2CC2)s1)C3 19072,c1(C(C)C)ncsc1C(=O)NCC1CCN(C(=O)C(F)(F)Sc2cnn(C)c2)C1 19073,CCC(CC(=O)NC(C)(Cc1ccccc1)C(F)F)c1ccccc1 19074,N1(C(=O)NCc2ccc(C3(C)NC(=O)NC3=O)cc2)CC=C(C(F)(F)F)CC1 19075,C(CCCCC(=O)NCC1CC=CCO1)N(C(C(C1CC1)OCC)=O)C 19076,N1(C(CC(=O)N=C2CC2)=O)CCCCCCC1C(=O)NC1(C(O)CO)CC1 19077,N1(C(CCSCC(C)C)=O)CCC(C)(NCC2CCC2CF)C1 19078,OCCC(N=c1nc(N2CCCC3(CC(O)C3)C2)c2[nH]ccc2[nH]1)C1CC1 19079,C(c1ccccc1Cl)=CC(=O)NCCCC(C)(C)NC(C1C(C)C1C)=O 19080,N1(C(C2CCN(C)C2=O)=O)CC2CCC2(CC(N2CCC3CCCC23)=O)C1 19081,c1(C(N2CCC(N(C)C(C3CC(C)(C)CN3C)=O)CC2)=O)nccc2[nH]ccc12 19082,N1(C(c2c(C)cncc2)=O)CCN(C(=O)COc2cccc(O)c2)CC1C 19083,c1(OC)ccccc1OC1CN(C(=O)C(F)=C(C)C)C1.C(c1ccsc1)=CC=O 19084,c1(NC(C2N(C(C3CCC(=O)NC3)=O)CC(O)C2)=O)nc(Br)ccc1[N+](=O)[O-] 19085,Cc1nc(C(N2CCC(C)(NC(C3CC4C=CC3C4)=O)C2)=O)c2ccccn12 19086,N1(C(C2C(CC(C)C)C2)=O)CCCC12CCN(C(=O)Cn1nc(O)ccc1=O)CC2 19087,N1(C(c2c(CC)ocn2)=O)CC(C)N(C(=O)CCCn2cnc(C#N)n2)CC1C 19088,c1(C(N2CCC(NC(C3(C)C(CC)CCC3)=O)C(F)C2)=O)cc2ccccc2[nH]1 19089,C1(CNC(C(C)=C(C)C)=O)CCN(C(C2CNC(=O)N2)=O)C12CCC2 19090,c1(OC)ccc(C(F)F)cc1C(=O)NC1CC(O)CN(C(=O)CSC(F)(F)F)C1 19091,c1(C(N(CC#C)CCO)=O)ccc(OCCOC)cn1 19092,CCC(C)C(C(=O)NCC1CN(C(=O)Cn2ccnc2C(C)C)C1)NS(C)(=O)=O 19093,CC1CN(C(=O)CC2COCCN2Cc2cc[nH]c2)CCC1=O 19094,CC(C)C(CNC(=O)CCC(C)(C)F)C(=O)Nc1cn(C)nc1O 19095,C(CC(C)CO)N(C(C(n1cc(CC2(O)CC(C(=O)O)C2)nn1)C)=O)CCF 19096,N1(S(CC(C)C)(=O)=O)CC2(CCN(Cc3ccccc3C(=O)O)C2)C1 19097,c1(C(=O)NCC2N(C(C(C)n3cccn3)=O)CC(O)C2)cncc2ccccc12 19098,C1(C(N2CCN(C(C(C(=O)OCC)(C)C)=O)CC2C)=O)CCn2ncnc2C1 19099,N1(C(C(C)(F)F)=O)CCOC2(CCN(C(=O)C=Cc3c(F)ccc(Cl)c3F)C2)C1 19100,N1(C(c2cnccn2)C(=O)NCCCC)CCC(C(N)=O)C(C(C)C)C1 19101,c1(N2CC3C(N(C)C)C3C2)nc(=NCC2(C3CCC3)CC2)[nH]c2c1SCC2 19102,N1(C(CSCC#C)=O)CCC(C)(C(=O)NC(C)(C)CCOC)C1 19103,C(C(=O)NCC1CCCC1NC(c1nccn1C(C)C)=O)(C(C)C)n1ncc(C)c1 19104,c1(C(=O)NC(CC)CN(C(=O)C(O)C2CC2)C)cn(C(C)(C)C)cn1 19105,CN1CCn2ncc(C(=O)NC3CC4CCC(C3)N4C(C3(C)CC3)=O)c2C1 19106,N1(C(C(C)SC(C)C)=O)CC2(C(=O)OCC3CC4(CCC4)C3)CCC1CC2 19107,c1(CNC(C(C)SC(F)(F)F)=O)cccnc1CNC(c1cc(Cl)cn1C)=O 19108,N1(CC(=O)Nc2coc(C(F)F)n2)CCC(CNC(C2CCCC2(F)F)=O)CC1 19109,c1(CNC(c2cc(C(C)(C)C)on2)=O)c(F)cc(Br)cc1F 19110,c1(C(C)=O)cc(=NCC(C2CC2)NC(=O)Cc2ccc(Cl)nc2)[nH]cc1[N+](=O)[O-] 19111,c1(CNCc2nc(CN=c3c(C(C)C)c[nH][nH]3)sc2)cc(Br)cnc1Cl 19112,C1(CC(=O)NCC(CN(C(C2CC(=O)C2)=O)CC)O)CCNC1=O 19113,CCC(C)(C)C(O)C(=O)NCC#CCNC(C1CCC2(CC1)CC2)=O 19114,N1(C(CC(CC)SC)=O)CC2CN(C(C3(OC(C)C)CC3)=O)CC(C1)O2 19115,c1(NC(c2csc(C(=O)Nc3ccccc3I)n2)=O)ccc2c(c1)COC2 19116,N1(C(C(C)n2cccc2)=O)CC2CC1(C(=O)NC1CCOC1(C)C)C2 19117,C(=O)(C(C)CS(C)(=O)=O)NC1CC(NC(c2ccc(-n3ccc(C)c3)cc2)=O)C1 19118,C1(C(=O)NCC2CN(C(C(=O)N(C)C)=O)CC23CCC3)CCc2cnn(C)c2C1 19119,c1(C(=O)NC2CCN(C(=O)CSC(F)(F)F)C2)cc(F)c(F)c(F)c1 19120,C(=O)(C1=CCCN(Cc2ccc(Cl)c(I)c2)C1)Nc1cc(C(=O)OC)cc(F)c1 19121,c1(C(CC)C(=O)NCc2cc[nH]c3nccc2-3)cccc2ccccc12 19122,C1(C(C)(C)NC(COCCC=C)=O)CCN(C(=O)C(C2CCCCCC2)C)CC1 19123,c1(C(=O)OC(c2ccncc2)C(=O)OCC)cscc1OC 19124,N1(C(C(C(C)C)NC=O)=O)C2CCC1CN(C(=O)CN1CC=CC1)CC2 19125,N1(S(CCC)(=O)=O)CCN(C(c2cc(C(C)C)ccc2Br)=O)CC1COC 19126,N1(C(CC(CNC(=O)C#CC(C)(C)O)OC)=O)CC2(CCNC(=O)O2)C1 19127,C#Cc1ccc(CNC(C2CCCCN(C(C3CCC(CC)C3)=O)C2)=O)cc1 19128,c1(SCC)ccccc1CC(=O)NCC1(NC(C2(O)CCSC2)=O)CCCCC1 19129,N1(CCNC(C(CNC(C2(F)CC2)=O)N(C)C)=O)CCNC(=O)C1 19130,c1(C2(C(=O)NCCCN(C(CCC=C)=O)C3CC3)CCC2)ncccc1F 19131,Cn1c(-c2ncccc2C(=O)Nc2ncc[nH]2)cc2ccccc12 19132,C1(C(N(C)Cc2nnnn2C)=O)N(C(C2CCCN2C2CC2)=O)CC12CCCC2 19133,C(=O)(CC(C)CCCCCCCCC)NCC(C1CCC1)NC(C(F)=CCC)=O 19134,C(c1cc(Br)cs1)=CC(=O)NC1CCCN(C(C2CCNC2=O)=O)C1 19135,N(C1COc2ccc(Cl)cc21)C(C1C2CN(C(c3ncccn3)=O)CC21)=O 19136,Cc1ccc(F)c(CNC(C2(C)CCCN(C(=O)C(C)OCCN(C)C)C2)=O)c1 19137,C(C)(CCCCNC(c1cccc(Br)c1)=O)NC(c1cc(C)ns1)=O 19138,C(CCCCCCCO)=CC(N1C(C2(O)CN(C(=O)C3=CCCO3)C2)CCC1)=O 19139,C(=O)(CCS(=O)(=O)Cc1ccccc1)N(CCCNC(C1C(C)C1)=O)C 19140,c1(CC)nc(C)c(C(=O)NCC2(CCNC(=O)C(C(C)C)NC=O)CC2)o1 19141,c1(C(=O)NC)cc(C)[nH]c(=NCC(C)(C2CC2)NC(=O)CCN(C)C(C)=O)n1 19142,C1(C)(NC(CC=C=C)=O)CCN(C(=O)CC(C)C)CC1 19143,c1(C(N2CCC(N(C(c3cc(C)c(O)cc3)=O)C)C2)=O)ccc2nc(O)[nH]c2n1 19144,c1(OCCC(=O)NCC2CC(NC(C3N(C(C)C)CCC3)=O)C2)cccc(F)c1 19145,CCCC(C)(O)CC(=O)N1CC2(C1)CN(c1ccc([N+](=O)[O-])cc1)C2 19146,N1(C(c2ccc(C)o2)=O)CCN(C(=O)C=CCN2CCCC2)C(CCO)C1 19147,N1(C(C=CC2CCN(C(CCOCC(C)(C)C)=O)CC2)=O)CCCC(N=[N+]=[N-])C1 19148,c1(C(N2C(CC(=O)NC)CN(C(=O)C(F)OC)CC2)=O)cc(C)c(C)cc1C 19149,CC1CCCN(CCNC(=O)CC2CCN(C(C3(C)CNC(=O)N3)=O)C2)C1 19150,N1(C(c2ccc(C(C)(C)C)[nH]2)=O)CC2CCCC2(Nc2ccnc3ncnn23)C1 19151,c1(NCCc2cc(Cl)no2)nc2ccccc2nc1N1CC2(CCC2)CC1CO 19152,c1(C(N2CCC(CNC(C(C=CC)O)=O)C(C)C2)=O)cc(C)cc(OC)c1O 19153,N1(C(C(CC=C)C)=O)CC(CN(C)C(c2cc(C(C)(C)O)on2)=O)C2(CC2)C1 19154,O=C1CCC(C(=O)N(CCC(N2CCC(F)CC2)=O)C2CC2)CC1 19155,C12(C(N3CC(C(C)NC(C45CCN(CC4)CC5)=O)C3)=O)CCCCC1C2(F)F 19156,c1(N2CCC(SC)CC2)ccnc2c1CCCC2O 19157,N1(C(c2cn(Cc3cnns3)nn2)C)CCN(C(=O)CCc2cnc[nH]2)CC1 19158,CCC(c1cccc(Cl)c1)=CC(=O)NC1CCC1NC(c1ncoc1C1CC1)=O 19159,C12(CNC(c3cc(C)c(C)o3)=O)CCCCC1CN(C(c1ccc[n+]([O-])c1)=O)C2 19160,C#CCCCCCCC(=O)NCC1(O)CCN(C(=O)CCC2CCCCC2)CC1 19161,C(CCCCC(=O)N(C(CNC(c1ccncc1C)=O)C1CC1)C)OC 19162,N1(C(c2c(C)[nH]nc2C(F)(F)F)=O)CC2CCN(C(C3CC3F)=O)CC(C2)C1 19163,C1(CCC(=O)NCCN(C(CC)C)C)CCCCN(CC2CC3(CC(=O)C3)C2)C1 19164,c1(NC(C2C=CCN2C(c2ccc(F)c(Cl)c2)=O)=O)cccc(F)c1Cl 19165,N1(C(Cc2cnc(C)s2)=O)CC2(CCC2NC(C2CCCC(=O)N2)=O)C1 19166,Cc1nc(CC(=O)NCC(O)CNC(=O)C(C)(C)CN(C)C)c(C)s1 19167,c1(C(=O)NCC2(C)CCN(C(C(C)OCC=C)=O)C2)ccc(OC)c(OC)n1 19168,c1(C(=O)NC2C(NC(Cc3ncc(C)o3)=O)C2)cncc(N)c1C 19169,n1(CC)nc(C(=O)NCC2COC(CNC(c3sncc3C)=O)C2)cc1O 19170,c1(CNC(=O)CC(C2CC2)NC(c2ccc(Cl)cc2)=O)cccc2[nH]ncc12 19171,N1(C(C=C(C)C(C)C)=O)CC2CN(C(=O)CC3CCC(C)(C)CC3)CC(C1)O2 19172,CC1(C)CCC(C)(NC(C2CCCCN2C(C2CCS2(=O)=O)=O)=O)CC1 19173,Cc1scc(CNC(C2(NC(C3CCC4CC34)=O)CCN(C)C2)=O)c1C 19174,N1(C(CSCC=C)=O)CC2CCC1CN2C(c1cc(CC(=O)OC)on1)=O 19175,C1(C2(O)CCOC2)(C(=O)NCC(CC)NC(C2CC2c2ccccc2F)=O)CC1 19176,C1(C(=O)NCC(C)CNC(=O)CCCN2CCCC2)CC(C)OC(C)C1 19177,CCC(C)CCC(=O)N1CC(O)CC1C(=O)NCC1(CCCO)CC1 19178,c1(C(=O)NCCC(C(=O)N(CC(CC)(C)OC)C)OC)cnn(C)c1C#N 19179,C1(NC(CC)=O)CCCC1C(=O)NC1(CO)CC(C)C1 19180,c1(OC)cc(C#N)ccc1C(=O)N(C)Cc1ccc(C)cn1 19181,C1(NC(C2(NC(C)=O)CCCC2)=O)CCCN(C(C2CC(=O)NC(=O)C2)=O)C1C 19182,Cc1n[nH]c(C)c1C(=O)NC(Cc1ccc(F)cc1)CC(=O)NCC1CCO1 19183,c1(C(N(C(CNC(=O)CC2CCSCC2)C2CC2)C)=O)cc(Cl)cnc1O 19184,c1(OC)ccc(C(=O)NCC2(NC(=O)C(C)=CC(C)(C)C)CCOC2)nc1Cl 19185,c1(CC)[nH]c(C(=O)NC2(C)CC(NC(=O)C(C)(O)CC)C2)nc1Cl 19186,Cc1ccc(F)c(C(N2CC3CC2C3NC(=O)C2=CCC2)=O)c1 19187,C1(C)(C(C[SH2]C)C)CCCN(C(C2(C(F)F)CC2)=O)C1.C1CC(=O)N1 19188,N1(C(C2CSCCN2C(=O)CN(CCO)CCO)=O)CCc2ccccc2C1 19189,c1(C(=O)NCCCOCCN(C(C(F)=C(C)C)=O)C)ccc(C(F)(F)F)s1 19190,N1(C(CNC(c2ccccc2Cl)C)=O)CC2OC(=O)N(C3CCOC3)C2C1 19191,Cc1c(NC(C2CC(C)CN2C(C2CCC(=O)N2)=O)=O)cc(Cl)cc1Br 19192,c1(C(C)C)nc(=NCC(C)N(C)C(c2ccc3ccnn3c2)=O)s[nH]1 19193,C1(NC(C(C)SCC)=O)CCC(C(=O)NC2CCC2C(=O)NC(N)=O)CC1 19194,c1(C(N(CCCNC(C2(C)CC(=C)C2)=O)C(C)C)=O)ccnc(C2CC2)c1 19195,N1(C(c2ccc(C)n2C)=O)CCN(C(c2n[nH]cc2F)=O)C(CS(C)(=O)=O)C1 19196,C(C#Cc1cn(CCCO)nn1)NC(=O)NOC1CCOCC1 19197,O=C(N=c1[nH]ccc2cc(Br)ccc12)C1CC2CC2N1C(c1ncccc1Cl)=O 19198,C1(NC(C=C2CCC(C)C2)=O)CCCCCCC1(C)C 19199,C(=O)(CCCC(F)F)NC(C1CCCCN1C(=O)Cc1cscn1)C 19200,c1(C(=O)NCCC(C)NC(=O)C=C(C2CC2)C2CC2)ccnc(N(C)C)c1 19201,N1(C(c2c(CC)ncs2)=O)CC2CC(C1)CN(C(=O)C(C)(C)CC)C2 19202,N1(C(c2cnc(=N)[nH]c2)=O)CCC2(CCC(CNC(C3CCCC3)=O)OC2)CC1 19203,C1(C(N2CCOC(c3ccc(C)s3)C2)C(=O)NCCC)CC2(CCCO2)C1 19204,NS(=O)(=O)N1CC(C(=O)NC2CCCN(C(C3CCN(C4CC4)S3(=O)=O)=O)C2)C1 19205,c1(CC)noc(C(=O)N(C2CN(C(c3cn(CC)nc3C)=O)C2)C)c1C 19206,C(=O)(C(C#N)C1CC1)N1CC(CCN(C(C)(C)C)C(=O)OCc2ccccc2)C1 19207,C1(CNC(CCOCCOC)=O)CN(C(=O)Cc2cnoc2)CCCO1 19208,c1(C(=O)NCC(C2(O)CN(C(C(C)OCC)=O)C2)(C)C)ccc(Cl)c(F)c1 19209,C1(CN(c2ccc(Br)cc2)C)CCC(=O)N(C(=O)CSC2CCOC2)C1 19210,N1(C(C2CC3(CC(NC(CC(C(C)C)C)=O)C3)C2)=O)CC2(CCCN2C)C1 19211,CC1CC(C)(C)N1C(=O)C=CCC(C)(C)NC(=O)CSC(C)(C)C 19212,c1(C(=O)NCC(C)N(C(Cc2cc(COC)on2)=O)C)ccn2c1CCCC2 19213,C(CCCCCNC(c1c[nH]nc1C1CC1)c1nnnn1CC1CCCO1)OC 19214,CC(c1ccccc1)=CC(=O)NCC1CC(NC(c2cc(Cl)nn2C)=O)C1(C)C 19215,C1(NC(=O)CCC2CC2(Cl)Cl)COCCN(C(=O)C2=CCC2)C1 19216,C(=O)(C(C(C)C)NC(=O)C(C)NC(C)=O)N1CC(C)(NC(C2(C)CC(=C)C2)=O)C1 19217,N1(C(c2c(CC)oc(C)c2)=O)CCN(C(=O)CC(C)(F)F)C2CCCCC2C1 19218,c1(SC)ccc(C(=O)NC2CCN(C(=O)CS(C)(=O)=O)C2C)cc1[N+](=O)[O-] 19219,CCC(C)(CC)C(=O)N1CCN(C(c2sc(C)nc2C)=O)C(CC(F)(F)F)C1 19220,C1(CC)CN(C(=O)C(C)C(C)NC(=O)CC2CNC(=O)O2)CC(=O)N1 19221,c1(C(N2CC3CC(CNC(C4(CC=C)CC4)=O)C3C2)=O)cc(OC)c(O)c(Cl)c1 19222,N1(C(C=CC)=O)CCC(C(=O)NC2CC(CO)C23CCC3)=C(F)C1 19223,c1(C(=O)NC(C)CNC(=O)CC2CCCCC2)cn(C(C)(C)C)nc1C(C)(C)C 19224,N1(C(c2c(C)ocn2)=O)CCN(C(C2CCC3(CCC3)C2)=O)C(C(C)C)C1 19225,CC1CCC(CO)N1C(=O)NCCCC(C)(C)C 19226,C1(N(C)C(c2ccncc2O)=O)CCN(C(c2cnc(-c3ccoc3)s2)=O)CC1 19227,Cc1c(C(=O)NC2CCC(CNC(c3ncc[nH]3)=O)C2)cnn1CC(C)(C)O 19228,Cc1nc2c(C)cc(C(=O)N(C(CO)CC(C)C)C)cn2n1 19229,c1(C(N2CC(C)C(NC(c3c(F)ccc(O)c3O)=O)C2)=O)cccc(S(C)=O)c1 19230,C1(C(=O)NCc2ccc(C(C)NC(=O)CSC3CC3)cc2)CC(F)(F)C1(C)C 19231,N1(C(c2c(CCC)[nH]cc2)=O)CCC2(CCC2)C(NC(=O)CCS(N)(=O)=O)C1 19232,CCC(CC1CCCC1)C(=O)N1CC(COC)(NC(=O)Cc2nonc2C)C1 19233,c1(C(N2CCC(N(C(C(C(C)OC)O)=O)C)CC2)=O)cn2ccccc2n1 19234,CC1CCC(CNC(=O)C(C)(C)n2cccn2)N(C(=O)CC2COCC2(C)C)C1 19235,C(=O)(CCCCCC#N)NC1CCCN(C(c2c(C)noc2C(F)F)=O)C1 19236,C(=O)(C1COc2ccccc21)N1CC(CN(C(C(C)OCC2CCCO2)=O)C)C1 19237,C1(CC(=O)NCCC(C)N(CCC)C)CCN(C(c2cscc2C)=O)C1 19238,c1(CNC(=O)NC(C#C)CC2CCC2)c(F)cc(Cl)cc1Cl 19239,C1(C(F)F)(CNC(C(C)O)=O)CCN(C(=O)CCN(S(C)(=O)=O)C)C1 19240,N1(C(C)C)CCN(C(=O)C(CCF)NC(C2CCC(C(N)=O)C2)=O)CC1 19241,C(=O)(CC(C)(C)C)NC(C1CCN(C(c2cnc(C(=O)O)[nH]2)=O)CC1)C 19242,[N-]=[N+]=NCCCCCC(=O)NC1CCCC(NC(=O)CC(F)(F)F)CC1 19243,C1(NC(C2(NC(C3C=CCC3)=O)C(C)C2)=O)CC2(CCC2)C1 19244,CCC(CC)(CO)NC(c1cncc(CNC(C2CCN(CC)C2)=O)c1)=O 19245,CCCC(O)(CCC)CC(=O)N1CCC(NC(c2ccc3nccn3c2)=O)C1 19246,N1(C(C)=O)CC(C(N(C)CC)=O)C2(CC2)C1.C(CC(C)C)OCCN(CC)CC 19247,C(=O)(C(CCC)c1ccc(Cl)cc1)N(CC(C)NC(C=C(CCC)C)=O)CC 19248,C#CC12CCN(C1)NC2=O.C(C(C)(F)C(C)(C)F)NC(=O)CN(CC(C)(C)C)C 19249,C1(N(c2ncc(Br)cn2)C(C2CCCO2)=O)CC2CCC(C1)N2 19250,C(=O)(C(F)C1=CCCCC1)N1CCC(O)(C(C)NC(C2C(CC)C2)=O)CC1 19251,c1(NC(C2CCC(C)CC2)CC)nc2ccccc2nc1NCc1cccnc1 19252,C1(=O)NNc2ccc(cc2)S(=O)(=O)CN1.c1(OCCC)ccccc1C(F)(F)F 19253,C(c1ccoc1)=CC(=O)N(CC(Cc1ccccc1)NC(C1C(C=C)C1)=O)C 19254,C1(N(C(C(c2ccccc2)NC(C2CCC(=C)CC2)=O)=O)C)CCCC(C)(C)C1 19255,c1(C(=O)NCc2cc(C)ncn2)coc2c1CN(C(=O)C(c1ccccc1)C)C2 19256,C(=O)(CC(CNC(C1C=CCS1)=O)OC)NC1CCN(CC)C1 19257,C(Cc1ccoc1)(C(=O)NCCS(N)(=O)=O)NC(C(C)SCCCC)=O 19258,C(CCCCCNCCCCn1cc(C2(C)CCOCC2)nn1)OCC 19259,C(C(C(C)C)NC(c1ocnc1C(C)C)=O)NC(C(=O)NCCOC)=O 19260,C(=O)(C(CC)NC(C)=O)CSCC(CC)NC(=O)CC1(N(C)C)CC1 19261,C=C(Br)CC(C)(C)C(=O)NC1CCCCN(C(c2cc(COC)on2)=O)C1 19262,c1(C(=O)NCCN(C(=O)Cc2cc[nH]n2)CC)cc(C(C)=O)cs1 19263,C(CCC1CCC1)(C(=O)NCCc1ccon1)NC(c1cc(CO)on1)=O 19264,c1(C(=O)NCC(C)(CO)NC(c2nc(Br)c[nH]2)=O)c(F)cc(F)cc1F 19265,C1(C2CC2)(NC(C(C2CC2)SC)=O)CCN(C(=O)Cc2cc(C)ccc2F)C1 19266,c1(COC)nc(NCCC2COC(C)(C)C2)cc(=NC2CCC(F)(F)C2)[nH]1 19267,CN1CC(NC(C2(C)CCCN(C(C3CN4CCN3CC4)=O)C2)=O)C2(CC2)C1=O 19268,CC1=C(C(=O)N2CC3=C(C2)CN(C(c2c(C)ncn2C)=O)C3)C(=O)OC1(C)C 19269,N1(C(CCCC(C)=O)=O)CC(C)CN(C(=O)Cc2cc[nH]n2)C(C)C1 19270,c1(C(=O)NC2CC(N(C)C)C23CCC3)cccc(-c2csc(C(=O)O)n2)c1F 19271,C1(CNC(C2(C(C)(F)F)CC2)=O)(NC(C2CCCCS2(=O)=O)=O)CCCCCC1 19272,C#CC1(C(=O)N(C(C)CCCC)C)CCN(C(C2CCC(OC)C2)=O)CC1 19273,C1(NC(C(C)(C)CF)=O)CCN(C(=O)Cn2ccccc2=O)CCC1CO 19274,CC1CC(NC(=O)Cc2cc(C(F)(F)F)n[nH]2)CCN1C(=O)CC1CCC2CC12 19275,CCC(CNc1ncccc1C)CCO 19276,c1(C(=O)NC(C)(CNC(=O)C=CC(F)(F)F)C2CCC2)csc(C2CC2)n1 19277,N1(C(C(COCC)C)=O)CCC2CN(C(=O)C=CC3CCCN3C)C2C1 19278,c1(C(=O)NCC2CCCC(NC(c3cc(C)ns3)=O)C2)nccc(C)c1N 19279,CCCC(C)CCNC(C1CCOCC1NC(C1CCC1(OC)OC)=O)=O 19280,Cn1cnc(CNC(=O)CC2CCN2C(C2CCCC2)=O)n1 19281,c1(-c2n(C(C)CCN3CCCC3=O)ccn2)ccc(CC2CCN(C)C2)cc1 19282,C(=O)(C(C(C)(C)C)NC(=O)C(O)Cn1cncn1)N1CC(S(C)=O)C1 19283,CCC(C)(CNC(C1(NC(=O)CC2CCCOC2)CC1)=O)CC 19284,c1(NC(Cc2nccc(CC)c2)=O)ccc2c(c1)CCC2N(C)C 19285,C12(C(=O)NC(c3nnc(O)o3)C)CC(CO1)N(C(C1(CO)CCC1)=O)C2 19286,C1(C(N(C)CC2(N(C)C)CCC2)=O)CC12CCCCC2.C1(=O)C(C)(C)CN1 19287,Cc1ccc(C(=O)NC2CC(N(C(=O)CC(C)C3CC3)C)C2)c(O)c1C 19288,C(=O)(C1=NOC(C)(CNc2cccc(OCC(=O)O)c2)C1)OC 19289,c1(NC)c(C(=O)NC2CC3(NC(=O)C#CC4(C)CC4)COC2C3)cccc1F 19290,c1(NC(c2n(CC)ccn2)C)[nH]c(=NCCCn2cccn2)nc2ncn(C)c12 19291,Cc1nc(C2CC2)ccc1C(=O)NCC1CN(C(=O)C(F)C(F)(F)F)CCC1C 19292,C(CCN(C)C)(CN=c1[nH]c(=NCc2csnn2)[nH]c2cc[nH]c12)OCC 19293,N1(C(COC(C)C)=O)CC2CN(C(=O)Cn3nc(Cl)ccc3=O)CC2C1 19294,c1(C(=O)NCCOCCNC(C(C)NS(CC)(=O)=O)=O)ccc(C(C)=O)cc1F 19295,C1(c2cn(CC3C(CC(N4CCCOCC4)=O)CCC3)nn2)CCCS(=O)(=O)C1 19296,C1(C(=O)NC2(CO)CN(C(CC3(C)CC3F)=O)C2)CC2(C1)CC1(CCC1)C2 19297,C(=O)(CCC(=O)NN(C)C)N1C(CNC(c2ncn(C(C)C)c2)=O)CC(O)C1 19298,N1(C(CC2N(CC)CCC2)=O)CCOCC(C(=O)NCCS(N)(=O)=O)C1 19299,C1(C)(C(N(CCCOC)CCO)=O)C=CCN1C(=O)C(C)=C1CCC1 19300,c1(C(=O)NC(C(C)C)CCN(C)C(c2coc(Cl)n2)=O)cc(F)ccc1N 19301,c1(C2C(C(=O)Nc3c(C)cnc(C(F)(F)F)c3)C2)cccc(Cl)c1[N+](=O)[O-] 19302,C1(CNC(c2nn(CC)c(C)c2)=O)CN(C(C2COC(C)(C)CO2)=O)CCN1C 19303,N1(C(c2c(C)cc(C)nc2)=O)C2COCC1CC(NC(C1(F)CC=CCC1)=O)C2 19304,c1(C(=O)NCC2N(C(C(C(C)C)C)=O)CCC2)ccn(C(=O)OC(C)(C)C)n1 19305,C1(NC(c2cnc(F)c(Cl)c2)=O)CCC2CCN(C(c3nocc3Cl)=O)C1C2 19306,Cc1ccc(Cl)c(C(=O)NC2CC(CNC(=O)Cc3nccn3C)C2)c1N 19307,C1(C(=O)N(C)CCN(C)C(C23CC(CC(F)F)(C2)C3)=O)(OC)CCS(=O)(=O)C1 19308,CC1CCc2sc(C(N3CC4CCCC3C4CNC(=O)C(C)C)=O)cc2C1 19309,C12(C(=O)NCCC(C)N(C(=O)C(C)OC3CCCC3)C)C=CC(CC1)C2 19310,N1(C(C=CC(C)(C)NC(c2c(C)n(C)nn2)=O)=O)CCC(C)C2(CCC2)C1 19311,C1(C(C)NC(C(C)OCCCC)=O)CCCN(C(c2cccs2)=O)C1 19312,c1(C(N(C2CCCCC2)CCNC(C(C2CCOC2)OC)=O)=O)c(C)ccn1C 19313,C1(NC(C2CCC=CCCC2)=O)CCC2CN(Cc3ccncc3Cl)CC2C1 19314,C(CN=c1nc(C2CCCC2)[nH]s1)C1CN(C(CCNC(C)=O)=O)C1 19315,c1(C(=O)NC2(C)CN(C(=O)C=CS(C)=O)C2)ccc(F)c2ccoc12 19316,N(C(=NCCC12CCC(C)(C1)OC2)NCC1(F)CCCCC1)CCSC 19317,C1(C(C)(C)C)CCC(NCC2(C(F)(F)F)CCC(N)C2)CC1 19318,c1(OC)ccc2cc(C(=O)NCC3CN(C(=O)C(C)S(C)(=O)=O)CCO3)[nH]c2n1 19319,C1(NC(c2c(CC)nn(C)c2)=O)CC2CCC1CC2NC(c1sccc1SC)=O 19320,c1(NC2CC(C)C2)cc(N2CCOC(CNC(C)=O)C2)ncn1 19321,CC(C)C(C(C)NC(c1csc(Cl)c1)=O)NC(c1sccc1CC#N)=O 19322,C=CC1COCC1NC(=O)CN(C(=O)C(C)(C)CC)C1CCC1 19323,c1(C(=O)NCCNC(C(C2CC2)OC)C)n[nH]cc1C1CCC1 19324,N1(C(C2CCC(CC)CC2)=O)CCCC2(CCC2NC(=O)Cc2cnn(C)c2)C1 19325,CCCCCCCCC(=O)NCc1ccoc1C(=O)NCc1snnc1C 19326,c1(-c2onc(COC(C)C)n2)ccc(OC(F)F)c(Cl)c1 19327,N1(CC(=O)NC2CCC(N(C(c3cncc(CC)c3)=O)C)C2)CCC(=O)NC1=O 19328,c1(CN2C(C(=O)Nc3ncn(C)c3)CC3CC32)cccc([N+](=O)[O-])c1F 19329,C1(CNC(Cc2c(C)scc2)=O)CCCC(CNC(=O)C(F)=CCCF)C1 19330,c1(C(=O)NCCCCC2CN(C(C3CC4(C3)CC4F)=O)C2)ccc(CO)cc1F 19331,c1(CC)cc(C(=O)NC(C)(C(=O)NCCCCN(C)C)C2CCC2)no1 19332,N1(C(C(CC)F)=O)CCC(C)C(NC(c2ccn(C3CCC3)n2)=O)C1 19333,C1(NC(c2cc(C)c(C)o2)=O)CCC2CC1CN2c1nnc(C(N)=O)s1 19334,C1(O)(CNC(C(C)OCCN(C)C)=O)CCCN(C(c2ncccc2N)=O)CC1 19335,C(=O)(C(F)C(F)(F)F)NC(c1c(CC)cccc1)CNC(=O)CC(=O)NC 19336,C(=O)(NNc1cc(F)c(F)c(F)c1)c1n(CCN)ncn1 19337,CC1CCN(C(=O)CC2(N(C(=O)C3=CCC(C)CC3)C)CC2)CC1(C)C 19338,C12(C(N3CC(C(C)C)C3)=O)CC(C)(CN1C(C1NC(=O)OC1C)=O)C2 19339,N1(C(C2(C)C=CCC2)=O)CCN(C(C23CCC(CC2)OC3)=O)CC12CCC2 19340,S(=O)(=O)(c1cccc(=NCC2(C3CCCO3)CCC2)[nH]1)NC(CC)CN(C)C 19341,CCC(CC)C(=O)N1CC(NC(C2(Cc3cccc(F)c3)CC2)=O)C(C)C1 19342,C(=O)(CCCC#N)NCC(CC)N(C(=O)C(N1CCCC1)C1CC1)C 19343,C(=O)(C(C)C(C)(F)F)NCCC1CC(NC(c2c(CCC)n[nH]c2)=O)C1 19344,Cc1cc(C)c(C(=O)NCCOCCNC(=O)C(C)Cc2cnn(C)c2)c(Cl)n1 19345,CN1CCN(C(c2cccnc2)=O)CC1C(=O)N(C1CCCC1)C1CC1 19346,N1(C(CN(CCOC)C)=O)CC2CCC1C(NC(=O)C(C(C)(C)C)C1CCC1)C2 19347,Cc1ccccc1C1(C(=O)NCCC2CCCN2C(c2ccc(F)s2)=O)CCC1 19348,c1(C(=O)NCC2(C(=O)NCC(C3CC3)OC)CC3(CC3)C2)ncc2ccccn12 19349,Cc1noc(C(=O)NC2CC(OC(C)(C)C)C2)n1 19350,C1(c2c(CC)c(C)no2)CCN(c2cc(NCC3CC(C)N(C)C3)ncn2)CC1 19351,CS(=O)(=O)CCC(=O)N1CCC(C2OCCC2NC(=O)CO)CC1 19352,C1(NC(c2c(OC(C)C)cccc2)=O)CN(C(=O)CC2CCSCC2)CCC1F 19353,C(=O)(C(C)CNC(=O)C(Cn1ccnn1)NC(=O)CCn1cccc1)OC 19354,C(=O)(C1=C(C)OCCS1)NC1CC2CN(C(c3nn(C(CC)C)c(C)c3)=O)C1C2 19355,C(=O)(C(F)CCC(C)C)NC12C(NC(C3N(C(CC)=O)CSC3)=O)CC(CC1)C2 19356,C12(C(=O)NC(CC)COCC3CC3)CC1CCN2C(C1CN(C)C1)=O 19357,C1(C(=O)NCCC2(NC(c3c(OC)scc3)=O)CC2)CCCC(C(N)=O)C1 19358,N1(C(C#CC(=O)N(C)C)=O)CC=C(CCNC(C2(F)CCS(=O)(=O)C2)=O)CC1 19359,C(=O)(C1=CC(O)C(NC(c2cccc(CC)n2)=O)C1)NCC 19360,CCCC(CCCNC(=O)C=CBr)NC(=O)C(C1CC1)OCC 19361,CS(=O)c1cccc(C(N2CCN(C(=O)CCF)C3CCC23)=O)c1 19362,C(CC(C)(C)C)(C(=O)NCCOCCCNC(=O)CCCN(C)C)OC 19363,c1(C(=O)NCC(C)CNC(=O)CCc2cncs2)ccc2c(n1)NCC2 19364,C1(N(C(c2ccc(C3COC3)cc2)=O)CC)CCCN(C(c2cn[nH]c2)=O)CC1 19365,c1(C(=O)Nc2c(CN)nc[nH]2)ncc(S(=O)(=O)NC)n1CC1CC1 19366,c1(C(N(CCCNC(C(C2CCCC2)OCC)=O)C)=O)c(C)nn2ncccc12 19367,C1(NC(c2c(CCC)nns2)=O)CN(C(=O)C(C)S(N)(=O)=O)CC12CCC2 19368,N1(C(c2c(C)[nH]c(C(C)(C)C)c2)=O)CCC2(CC(NC(=O)CSC(C)C)CO2)C1 19369,C1(C(=O)NCCSC)CCC2(CN(C(C3CC4CCCCC4N3)=O)C2)O1 19370,c1(C(CC)C)nc(C)cc(=NC(=O)c2ccn3ncc(I)c3n2)[nH]1 19371,Cc1cc(C)c(CC(=O)NC2CC(N(C)C(c3ccc(C#N)[nH]3)=O)C2)s1 19372,c1(C(N2CC=C(CNC(C3CCOC3)=O)CC2)=O)ccc2nn[nH]c2c1 19373,C#CCCCCCCC(=O)NNC(=S)c1ccccc1N(C)C 19374,c1(OC)cccc(C)c1C1(C(=O)NC(c2cc(OC)ccc2F)C2CC2)CC1 19375,C#Cc1cn(C)nc1C(=O)NC(C)CC(=O)N(CC(N)=O)CC(N)=O 19376,c1(C(=O)Nc2c(C)cc(NC(c3coc(C#N)c3)=O)cc2)ccc(F)c(Cl)c1F 19377,N1(C(C2N(C(=O)OC(C)(C)C)C(C)CC2)=O)CC2CC(NC(C3(O)CC3)=O)C1C2 19378,Cc1nc2ccc(C(=O)NCC3CCCC3NC(=O)CC3CC3(Cl)Cl)cc2n1C 19379,N1(C(c2cnc(CCC)s2)=O)CCCC(CN(C(C)C(=O)NC)CCC)C1 19380,N1(C(CC(C)C(F)F)=O)CCC2CCN(C(c3cc(C(F)F)ccc3F)=O)CC12 19381,C1(C(N2CCN(CC)CC2)=O)CC12CCN(c1nnc(C)c(C)n1)CC2 19382,CC(C)(C)CC(O)CC(=O)NC1CCN(C(c2c(N)cccc2F)=O)CC1 19383,C1(NC(=O)CCC2CC2(Cl)Cl)(CO)CCCN(C(C2CCCNS2(=O)=O)=O)C1 19384,C1(CC=C)(C(=O)NCCC2CC3C=CC2C3)CCCN1C(C1CSC1)=O 19385,N12CC(O)CC1C2=O.C1(NC(=O)OC(C)(C)C)CC(NC(C2(Cl)CC2)=O)C1 19386,C1(NC(CC2ON=C(C)C2)=O)CCN(C(c2cc(C)ns2)=O)CC1CO 19387,N(C(C)=S1(=O)CCCC1)(N1CCC(C(C)C)C1)C(c1ccc(F)cc1F)=O 19388,c1(OC)ccc(C)c(C(N2CC(NC(=O)C(C)CSC)C(C)(C)C2)=O)c1 19389,C1(NC(C(C)C2CC2)=O)CN(C(=O)CCc2cccc(Cl)c2)CCC12CCC2 19390,Cc1cc(N)cnc1-c1nc(CC2N(Cc3ccccc3)CC2(C)C)no1 19391,C(=O)(C1=NOC(C)C1C)N1CCC(NC(c2cc(C(C)C)on2)=O)(CO)C1 19392,Cc1cnc(C(N2CCC(NC(c3cc(F)c[nH]3)=O)C(CO)C2)=O)c(C)c1 19393,CC(CC(C)(C)C)C(=O)NCc1cc(C(=O)NCCCC2CC2C)n[nH]1 19394,CC1CCN(C(C2C=CCC2)=O)CC1CNC(c1cnccc1Cl)=O 19395,C(=O)(C(C)(C)C(C)C)N(CC(CNC(Cc1ncc(C)o1)=O)O)C 19396,C(CCCCCNC(C1CCCN1C)=O)NC(C=CCCC=C(C)C)=O 19397,C(=O)(CCCCC(=O)N1CCC(NC(C2(C(F)F)CCOCC2)=O)C(O)C1)NC 19398,CC1CC(=O)NC(C(=O)NCC2(CNC(c3nocc3C3CC3)=O)CC2)C1 19399,N1(C(CN(C)C)=O)CCC2CN(C(=O)CCc3cnc(O)[nH]3)CCC2C1 19400,N1(C(C(C(C)C)OC)=O)CC(CNC(c2cccc3nn[nH]c23)=O)CC12CCC2 19401,C12(C(N3CCC(CNC(C(C(C)C)O)=O)C3)=O)CC3CC(CC1C3)C2 19402,c1(C(N(CCN(C(CSCC)=O)C(C)C)C)=O)nc(C)ncc1Cl 19403,N1(C(c2c(C)noc2N)=O)CCCC(NC(=O)CC(O)C2CCCC2)CC1 19404,C12(C(=O)NC3CCN(CC)C3=O)CC(CCO1)N(C(=O)Cc1cc(C)cs1)C2 19405,C(=O)(CC(=O)NC(C)CNC(=O)C(C)C1CCC1)NCC#C 19406,N1(C(C(C)NC(c2ccco2)=O)=O)CC2CCCC(NC(=O)C(C)(C)F)C2C1 19407,c1(C(=O)NC2CC(CNC(c3cnc(C)[nH]c3=N)=O)C2)nccc2ncccc12 19408,CC1CCCC(C(N2CCN(c3ccc(C(=O)O)cc3)CC2)=O)C1C 19409,CC1CN(C(c2ncc[nH]c2=O)=O)CC(CCNC(c2cn(C)nc2Cl)=O)O1 19410,C(=O)(CC(F)(F)C(F)F)NCC1(NC(CCNC(C2CCCCC2)=O)=O)CCC1 19411,C12(C(=O)NC(C3CCN(C(c4nc(C)sc4C)=O)CC3)CO)CC3CC1C2C3O 19412,N1(CC(=O)N(C(c2cn(Cc3nnc(C)o3)nn2)C)C)CCCC(C(C)O)C1 19413,C(=O)(CCC(=O)NN(C)C)N1CC(C2CC2)(C(=O)NC(C2CCCCO2)CC)C1 19414,Cc1cc(NC2CCOc3ccccc3C2)ncc1S(=O)(=O)N(C)Cc1ccns1 19415,C1(CC(=O)NCC2(NC(C3C(C(C)C)(CC)C3)=O)CCC2)(N(C)C)CCCC1 19416,c1(C(N2CCCC(CNC(CSC(C)(C)C)=O)C2)=O)cccc2nonc12 19417,N1(Cc2cccc(CCC=C)c2)CCS(=O)(=O)CCC1c1ccccc1 19418,N1(C(C2CC=CC(NC(C(CC)(C)O)=O)C2)=O)CC=C(CO)CC1 19419,C(=O)(C(CO)NC(=O)C(F)(F)F)NCC(CC)NC(c1ccn(CCOC)n1)=O 19420,C1(NC(C2(CNC(=O)CN(c3ccccc3)C)CC(=C)C2)=O)CCCCCC1 19421,c1(C(=O)NCC2CCCC(NC(C(C)c3cccs3)=O)C2)ccc2nccn2n1 19422,C=CCC(C(=O)NCC1CC2CCC(C1)N2C(=O)C=NOC)C(C)(C)C 19423,C12(NC(CCC=C=C)=O)CCCC(CN(C(C3CCCN3C)=O)C1)C2 19424,C(C)(CNC(c1ccc(-c2nncn2C2CC2)cc1)=O)(C(C)C)NC(C)=O 19425,C#CCCC(O)C(=O)NCCNC(C1CCC(Cc2cccc(Cl)c2)C1)=O 19426,CC(C)(C(=O)NC(CNC(=O)C(C)(C)n1cnnn1)CC(F)(F)F)C(F)(F)F 19427,CC1(C(=O)NCCc2n[nH]cc2C(=O)NCCC2CC(O)C2)CCCC1O 19428,N1(C(c2c(F)ccc(C)c2)=O)CCC2(CCCN2C(C2CSCCS2)=O)C1 19429,N1(C(Cc2ncc(C)o2)=O)CCC2(CCCC2NC(C2C=CC=CC=C2)=O)CC1 19430,CC(C)C(CC(=O)NCCCc1ccsc1)NC(c1c[nH]nc1C(F)F)=O 19431,C(C(C)(C)C(=O)NC1C2CN(C(C3CCCN3C(C)=O)=O)CC12)NC(C)=O 19432,c1(-c2cn(C3CC(C(C)OC)C3)nn2)cc(F)c(F)c(F)c1 19433,C(C(=O)NCc1ccoc1C(=O)NCC1CC=CCC1)(C(C)(C)C)OC 19434,CCCC(C)C(=O)N(C(C)(C(=O)NCc1nccc(OCC)n1)C1CC1)C 19435,C1(C(C)C)COCCN(C(c2sccc2CNC(=O)CC(F)(F)F)=O)C1 19436,N1(C(C2CCCN(C(C)=O)C2)=O)CCCC2CN(CCC3CCCCCC3)CC12 19437,C(=O)(C(F)CC(C)(C)NC(=O)C=CC(C)CC)NC1C(C=C)OCC1 19438,C1(N(CCC)C(c2[nH]cnc2C)=O)CCN(c2nnc(C3CC3)o2)CC1 19439,c1(N2C(C)CN(C(c3cc(=O)cc(Cl)[nH]3)=O)CC2)ncc(C#N)cc1Br 19440,c1(C(=O)NCC(C)NC(c2c(F)ccc(F)c2O)=O)c(F)ccc2nc[nH]c12 19441,C1(CN(C(CCn2c(C)ncc2)=O)C)CN(C(=O)C(N)=O)CC12CC2 19442,c1(-n2c(C(C(C)(C)OCCO)NC3CC(SC)C3)nnn2)cccc([N+](=O)[O-])c1 19443,C(CC(C)(C)NC(=O)CCOCC1CCC1)=CC(=O)N(CCCC#C)C 19444,C1(C)(CNC(C(C2CCN(C(c3coc(C4CC4)n3)=O)C2)C)=O)CCCOC1 19445,Cc1cc(CC(N2CCC(F)C(NC(c3ccoc3Cl)=O)C2)=O)ccc1CO 19446,N1(C(c2c(C)ccs2)=O)CC2CCC(NC(c3ccc4n[nH]cc4c3)=O)(C2)C1 19447,C(=O)(CCC(=O)C1CC1c1cn(C(C)C(=O)NC(C)(C)C)nn1)N(C(C)C)C 19448,CC(C(=O)NCc1cn(C2CN(C(c3ncccc3Cl)=O)C2)nn1)C(C)(F)F 19449,C12CCN(C1)C2=O.C1(C2CCCO2)(C(N(CC(=O)NC)C)=O)CCCC1 19450,C(=O)(C(C#N)C(C)(C)C)N1C(CC)CN(C(c2c(C)ncnc2O)=O)CC1 19451,C1(CNC(COC)=O)CCN(C(=O)C(C)COC)CC1C1CC1 19452,CN1CC2CCN(C(=O)C=CCN(C)C(C3CS(=O)C3)=O)CC2C1 19453,c1(C(=O)NC2CC(C)N(C(c3ocnc3C(F)F)=O)C2)ccc2c(c1)CCC2 19454,C(=O)(CS(=O)C(F)(F)F)NCC1CCCCN(C(CN(C)CCO)=O)C1 19455,CCCCCC(COC)C(C)NC(=S)NCCC(F)(F)F 19456,N1(C(C2N(C(C)(C)C)CC2)=O)CCCC2CN(C(=O)C3CC3)CC12 19457,N1(C(c2c(CC#N)cccc2)=O)CCCCC(NC(C23CC(CF)(CO2)C3)=O)C1 19458,C=CCC(CC(F)F)C(=O)NCC12CC1CN(C(c1cccc3ncnn13)=O)C2 19459,C1(C(N2CCN(C(CN(CC#C)C(=O)OC(C)(C)C)=O)CC2)=O)COCCNC1=O 19460,c1(C2(C(=O)N(C(CC)CF)CC)CC2)cccc(F)c1Br 19461,c1(C(N2C3(C(N)=O)CC3CCC2)=O)n[nH]c2c1CNCC2 19462,N1(C(CCC=C)=O)CC(C2CN(C(=O)C(c3ccccc3C)C3CCCC3)C2)C1 19463,CCC(CC(=O)NC1CCCC(NC(C2CC(O)CN2C(C)=O)=O)C1)C1CC1 19464,C(=O)(CC(C(F)(F)F)OC)NCC1C(CNC(C2(C(=O)OCC)CC23CC3)=O)C1 19465,c1(OCC)nccc(CNC(C2CC(C)CO2)=O)c1N.C(=O)(CS(=O)(=O)NC)NC 19466,C12(CNC(c3c(C(C)C)cccc3)=O)CCCC1CN(C(=O)C(C)N(C)C)C2 19467,c1(N(C)C)ncc(C(=O)NCC2CC(O)CN2C(c2ccc(O)nc2)=O)cc1Cl 19468,c1(CN(C(=O)NC2CCC(c3ccc(F)cc3)C2)CC)csc(C#N)c1 19469,N1(C(C(c2ccccc2)C)=O)CCN(C(=O)Cc2ccc(Br)cn2)C(CO)C1 19470,C(=O)(C1=COCCO1)NCC(C)(C1CCC1)NC(c1cc(CN(C)C)on1)=O 19471,C(=O)(C1=C(Cl)CCOC1)NCC1N(C(CCCCCN(C)C)=O)CC(O)C1 19472,Cc1nc(C)n(O)c1C(=O)NC1CCCN(C(=O)C(C)(C)C(N)=O)C1 19473,N1(C(CC(C)NC2(C)CCC2)=O)CCCC(CC(=O)N(C)C(=O)OC(C)(C)C)C1 19474,C1(C(N2CCC(C(C)CNC(=O)C(C)(C)F)CC2)=O)CC2(CCO1)CC2 19475,c1(OC)cc(C(=O)OCc2nc(C(C)OC)cs2)cnc1C(F)(F)F 19476,N1(C(C=CCN(C)C(c2ccc([N+](=O)[O-])o2)=O)=O)CCC2CCCCC2C1 19477,C1(NC(=O)C(C2CCOCC2)=O)CC(C(=O)NCC2CN3CCC2C3)CC1O 19478,Cc1ccc(C)c(CN(C(=O)CCCC(=O)c2cccs2)C2(C)CCCCO2)c1 19479,Cc1cc(C(N)=O)cc(C(=O)N(C)CCN(C(C2CCCC2(F)F)=O)C(C)C)c1 19480,N1(C(c2n[nH]cc2C2CC2)=O)CCC2(CC1)CN(CC1(N3CCCC3)CCC1)C2 19481,C=CCC(C)(C)C(=O)NC1CCC1NC(c1cccc(C(C)=O)c1)=O 19482,O=S(=O)(c1ccc(N2CCC3(C2)CC(F)(F)C3)c(Br)c1)NCC1CSCCS1 19483,C=CCC(C)(CC)C(=O)N1CCC(C)(CC(=O)NCCc2cc[nH]n2)C1 19484,N1(C(c2nccs2)=O)CCC(F)(C(=O)NCCCN2CCCC2=O)C1 19485,CC(O)(CNC(=O)C(C1CCC1)NC(c1cc(O)ccc1F)=O)C(F)(F)F 19486,N1(C(=O)CC2OCCCO2)CCC2CCCN(C(=O)Cc3ccoc3)C2C1 19487,C1(NCc2c(C(=O)NCc3cc(C(=O)OCC)no3)cco2)CCC(O)CN1C 19488,c1(OC)ncc(Cl)c(N2CCCC(NC(=O)CNC(=O)CC3CCCC3)C2C)n1 19489,N1(C(C(c2ccn(C)n2)C)=O)CC=CC(NC(=O)C(O)CCN(C)C)C1 19490,N1(C(c2c(C)nsc2)=O)CCC(C(C)NC(=O)CC2CCCO2)CC1 19491,Cn1nc(CO)c2c1CN(C(c1cc(-c3ccncc3)ns1)=O)CC2 19492,c1(C(N2CCC(OC)(CNC(=O)Cn3ncnn3)C2)=O)c(F)ccc(F)c1Cl 19493,C1(C(=O)NCCc2c(C(=O)NCCC(=O)NC)c[nH]n2)OCCOC1C 19494,O=C(CC1CCOC1)NOCC(=O)NCCOCCSc1nc[nH]n1 19495,C(C(C)(C)C(=O)NC1CNC(=O)OC1)N(C(C1C(C)CC1)=O)C 19496,O=S(=O)(c1ccc(Cl)c2cccnc12)N1CC(O)CC12CCS(=O)(=O)CC2 19497,C1(CC=C)(NC(=O)CC(C)F)CCCN(C(c2cc(C(F)F)ccc2Cl)=O)C1 19498,CC(C(=O)NCC1(O)CCCN(C(c2ccn3c2CSCC3)=O)C1)C1=CCCC1 19499,CC(C(=O)N1CCCC1CCNC(C1(C)CCC(=O)N1)=O)S(N)(=O)=O 19500,Cc1cccc(F)c1CC(=O)N(C)CCOCCNC(=O)CC1CCOC1C 19501,N1(C(CSCC#C)=O)CCC(NC(=O)C(C(C)C)n2cnnn2)C1C1CC1 19502,C(=O)(CC(C)CN(C)C)N1CCC(CN(CC)CC)C1.C(=O)CC(C)C 19503,c1(CN(CCNC(=O)CC2(C)CC2(Cl)Cl)CC)ccc(C)cc1C 19504,C1(C(=O)NCC(=C)Br)CC2CC1CN(C(=O)CCC1OCCO1)C2 19505,N1(C(C=C(C)C(C)(C)C)=O)CC(N=[N+]=[N-])CC1C(=O)NCc1cscn1 19506,N1(C(=O)CCc2cccs2)CCCN(C(C2CC3CC2CC3O)=O)CC1 19507,N1(C(C2(F)CCC(C)CC2)=O)CCOC2(C1)CN(C(=O)CCC1CC1(C)C)C2 19508,c1(OCC)ccc(C(=O)NCC2CN(C(c3ccnc(C)c3)=O)CC2C)cc1O 19509,C1(N(C(c2n(CC)ncn2)=O)C)CCCCN(C(=O)C=Cc2ccc(C)cn2)C1 19510,N1(C(C(Cc2cn(-c3c(C(=O)O)ccnc3)nn2)O)=O)CCNC(=O)C1C 19511,N1(C(CC=CC=C)=O)CCC(CNC(=O)CC(C(F)(F)F)OC)C(F)(F)C1 19512,CC1(NC(=O)CNC(N)=O)CCN(C(C2CCCC(F)(F)C2)=O)CC1 19513,C1(C(=O)NC(C(=O)NCCC(=O)NCC)Cc2cn[nH]c2)CCCCCCC1 19514,n1(CCC(=O)NC(CC(CC)=O)C(=O)O)ccc2ccc(F)cc12 19515,N1(C(CN(C(CNC(CC)=O)=O)C)=O)CC=CC(O)C1 19516,C(C(O)C(=O)N(CC(C)NC(=O)C(CN(C)C)N(C)C)C)=CCCC 19517,c1(C(=O)NC2CCC(C(=O)N(CCO)CC3CCCO3)CC2)nnc(O)cc1O 19518,c1(C(C)OC)nc(C)c(C(=O)N(C)CCNC(=O)C(=Cc2cccs2)C)s1 19519,CCC(CC)(CCNC(=O)CN1CCC(CO)CC1)NC(C1CCCCC1C)=O 19520,C(C)(CC(C)CC(C)C)(c1n(CC=C)nnn1)NCc1ccc(COC)o1 19521,c1(OCC)cc(NC2CCN(CC(=O)Nc3ccc(Cl)cn3)CC2)nc(C)n1 19522,C1(N(C(c2nc(C)sc2)=O)CC2CC2)CCN(C(=O)CC2(O)CCOC2)CC1 19523,Cc1nc(NCCC2CCCCN2C(C23CCCC(CO2)C3)=O)c(Cl)cc1C#N 19524,C1(CNC(COCCCC)=O)CC2(CCN(C(c3cc(C4CC4)ns3)=O)CC2)C1 19525,N1(CC(=O)N(CCCC)CCCC)CC2CCC(C(=O)NC3CCOC3)CC2C1 19526,c12nc(c(N)s1)C(=O)N(Cc1ccc(F)cc1)C2.c1(CCCC)cc(OC)no1 19527,c1(C(=O)NC2CC(NC(C3(c4ccn(C)c4)CC3)=O)C2)csc(S(N)(=O)=O)c1 19528,c1(C(C)=O)ncc(C(=O)NC2CCC(NC(=O)C(C)n3cnnn3)C2)s1 19529,C1(C(=O)NCC(C)CNC(=O)CC2COC(=O)N2)CCC12CCC2 19530,N1(C(C(C)C2CCCO2)=O)CCC2CCN(C(c3ccc(O)nn3)=O)CC2C1 19531,c1(C(C)C)nnc(C=CC(=O)NC2CCCCC2NC(=O)CCn2cccn2)o1 19532,Cc1cccc(C)c1NC(=O)C(N1CCCC(CC(=O)N(C)C)C1)CC1(C#N)CC1 19533,C(c1cc(Cl)ccc1Cl)=CC(N1CC(CNC(C2(COC)CCC2)=O)C2C1C2)=O 19534,c1(OC)ccc(C(N2CC(NC(=O)CC(C)OC)C(F)C2)=O)c(F)c1 19535,C(C)(CC(=O)N1C2CCC1CC(NC(C1(CF)CC1)=O)C2)(C(F)(F)F)N(C)C 19536,C(=O)(C(F)CC(C)(C)NC(c1ccc(O)cn1)=O)N1CCN(C)CC1 19537,C(C(C(=O)NCC(CC)NC(=O)C(c1cncn1C)O)c1ccccc1)OCC 19538,S(=O)(=O)(c1cnn(C)c1)N1CC(C(N2CCC(C(C#C)C)CC2)=O)C1 19539,S(=O)(=O)(c1cc(C)c(C)s1)NC(C1CCCN(CCOC)C1)C 19540,c1(OC)ncc(C)cc1-c1ccc(C2(NC(c3c(Cl)cnn3C)=O)CCC2)cc1 19541,N1(C(CCC#CC)=O)CCc2nc(CNC(c3cc4n(c3)CCCC4)=O)sc2C1 19542,C1(C(C)NC(c2conc2C2CCC2)=O)CCCN(C(c2cc(CO)cs2)=O)C1 19543,C1(C(=O)NCCC(=O)NC(CC(=O)NC(C)C)C)CC2(C1)CC(O)C2 19544,c1(CC)ccnc(C(N2CCN(C3CN(C(=O)C(F)CC4CC4)C3)CC2)=O)c1F 19545,N1(C(Cc2n(C)cnc2)=O)CCN(CCNC(N)=O)CC1 19546,c1(C(=O)NC(c2ccccc2F)CNC(C=CSC)=O)cccc2c1OCCN2 19547,C1(C2CCCN(C(=O)C3=CCCC3)C2)(NC(c2cc3cnccc3o2)=O)CC1 19548,c1(CC)nn(C)c(Cl)c1C(N1CCC(C)(CNC(C2CC23CCC3)=O)C1)=O 19549,c1(OC)ccn2ncc(C(=O)NCCOCC(F)(F)C(F)(F)F)c2c1 19550,C(C(=O)NCc1ccnc(O)c1)(C(C)C)NC(CN(C(C(C)C)=O)C)=O 19551,C12(NC(COC(C)C)=O)CCC(NC(c3cc(Cl)ncn3)=O)(CC1)C2 19552,CCC(CC(=O)N1CC(O)(CN(C)C(c2cc(C(N)=O)ccn2)=O)C1)C1CC1 19553,c1(C(=O)NCC2CCCCN(C(C(C=C)O)=O)CC2)c(C)nn2c(C)cccc12 19554,N12Cc3ccccc3C1C(=O)N1CC(C1)C2=O.C#Cc1nccnc1C(=O)OC 19555,C(C)(C)(CCCC(=O)N1C2CCCC1COC2)NC(C(CC)COC)=O 19556,S(=O)(=O)(c1ccc2ccccc2c1)N1CC2N(C(=O)C(F)Cl)C(COC2)C1 19557,N1(C(CC(C)OC)=O)CCC(NC(=O)CC23COCC(C2)C3)C1C 19558,C12(CC(=O)NCCCCCN(C(C3CC(SC)C3)=O)C)COCC(C1)C2 19559,C1(C(=O)NCC(CC(=O)NCCN2CCOCC2)OC)CCCCC1(C)C 19560,c1(C(N(C(CNC(C2(C)C(C(=O)OC)C2)=O)C)C)=O)cc(-c2ccncc2)on1 19561,C(=O)(C(C)CC(C)(F)F)NCC1(C(C)(C)O)CN(C(C=CSC)=O)C1 19562,C1(C(=O)NCCC(N)=O)C=CCN1C(=O)CC1COC(=O)C1 19563,Cc1cc(C(=O)NC2CCC2NC(=O)C=CBr)cc(Cl)c1Br 19564,c1(NC(=O)NC2C(CC)COC2)ccc(C)c(C(=O)OC)c1.C12(CC1)C(=O)N2 19565,C12(C(=O)NCCCC3(NC(C4C(C)OCC4)=O)CC3)CC3CC1C2C3 19566,C1(C(=O)NCc2ccc(-c3ccccc3)cc2F)CCn2c(O)nnc2C1 19567,C1(NC(CNC(=O)OC)=O)CCCCN(C(=O)CC2CN(C)CC2O)C1 19568,C(=O)(C(CC(C)C)C(N)=O)N1CCCC(O)(c2cn(Cc3c(C)sc(Br)n3)nn2)C1 19569,C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NCC(CNC(C1(C)CC(O)C1)=O)F 19570,N1(CC)CCOCC1C(=O)N(CC(C)(C)CNC(C1(COC)CC1(F)F)=O)C 19571,N1(C(c2n[nH]c(CC)c2Br)=O)CC(C)(C)CC1CNC(C1CCC1C)=O 19572,c1(C(C)C(=O)NCCCNC(=O)CC2NC(=O)NC2=O)ccc([N+](=O)[O-])cc1F 19573,N1(C(C2C=CCCC2)=O)CC2CC1(C(=O)Nc1ccccc1)C2 19574,C1(C(C(=O)NC)N(C2CC(n3cncn3)C2)C)CC2CCC1C2 19575,C(=O)(C1CCSc2ccccc21)N1CC(CNC(C(=O)NCC)=O)C(C)C1 19576,c1(CC(C)C(=O)NCCC2(O)CCN(C(=O)CC3(C#N)CC3)C2)cccc(F)c1 19577,Cc1ccoc1NC(C1CC1C(=O)Nc1cnns1)=O 19578,C1(C)(CNC(C(C)C2CCCC2)=O)CCN(C(=O)CC2SC(=N)NC2=O)CC1 19579,N1(C(CC(CC)C)=O)CCCCC2(CCN(C(c3ccccc3SCC)=O)C2)C1 19580,c1(C(=O)NCC2CN(C(C3C(C=C)C3)=O)C(C)(C)C2)cc(Cl)cc(Cl)c1O 19581,Cc1ccc(NC(CCNCC2CN(C(=O)OC(C)(C)C)CC2O)=O)cc1C 19582,C1(NC(C2=NNC(=O)C2)=O)CCCC2CN(C(C3CC=CC(O)C3)=O)CC12 19583,CC(C)CC(O)C(=O)NC(Cc1ccco1)C(=O)N(C)CC1(O)CCC1 19584,O=C(CCCCCCCO)NCC1CCCN1C(=O)Cc1cnc2[nH]ncc2c1 19585,C12(C(=O)NCCCCC)CCCC1CCN2C(c1ccc(CC)cn1)=O 19586,Cc1ccc(C(N2CC3(CCC3NC(=O)C(C)OCC3CC3)C2)=O)c(Br)c1 19587,C(=O)(CCC(CC)OC)NC1CCN(C(CCCC)=O)C1CC 19588,CCC(CC(F)F)C(=O)N1CCCC1CN(C)C(c1c(F)ccc(C)c1N)=O 19589,C1(CC)CN(c2ccccc2)CCN1C(c1cc(-c2ccccn2)[nH]n1)=O 19590,Cc1cc(C(=O)NC2(CN(C(=O)CN(C3CC3)C(C)C)C)CC2)c2ncccc2c1 19591,C=CCC(CC)N=c1[nH]c(N2CCC(OCCO)C2)nc2ncn(C)c12 19592,C1(C(=O)NCC(CO)NC(CCC=CC)=O)CCN(C(=O)C(C)(C)C)CC1 19593,C(=O)(C(F)(F)C(O)C(C)C)N1CCCCC(NC(c2c(C)nc(CCC)s2)=O)C1 19594,C1(CNC(CN(CCC#C)C)=O)CCOC1C(=O)N(C1CC(O)C1)C 19595,N1(C(=O)NC(c2nc(=O)[nH][nH]2)C)CCCC2(C=CCO2)CC1 19596,N1(C(CC(=C=C)C)=O)CCN(C(=O)C(C)Oc2ccc(Cl)c(Cl)c2)CC(O)C1 19597,c1(C(=O)OC)ccc(F)c(C(=O)NCC2CC(NC(=O)C(F)(F)C(C)O)C2)c1C 19598,C1(C(=O)NCC(C)(C)C(=O)N2CCOCC2CCO)CCCC(C#N)C1 19599,C1(NC(C2CC(=C3CC3)C2)=O)CCC2CN(C(=O)COc3ccncc3)CC12 19600,CC(C)C(Cc1ccccc1)C(=O)NCCC(C)N(C)C(c1cc(C#N)c[nH]1)=O 19601,c1(NC(C2CCC(NC(C=C(C)C(=O)O)=O)CC2)=O)cc(C#N)ccc1O 19602,C1(NC(c2c(CCC)n[nH]c2)=O)CN(C(C2C(C)(C)C2(C)C)=O)CCC1O 19603,CC1(CNC(N2CCC(C(=O)OC(C)(C)C)CC2)=O)OCCc2sccc21 19604,N1(CC)CC(C(N2CC3CC2C3NC(c2nccnc2N)=O)=O)CCC1=O 19605,c1(C(N2CCCCC2c2cccc(O)c2)=O)ccc(C2CC2)cc1I 19606,c1(C(=O)OCC)ccc(N(C2CCCN(C(c3cc(C(F)F)[nH]n3)=O)C2)C)nc1 19607,C1(CC(=O)N(CC(C)N(C(c2c(SC)ccs2)=O)C)C)CN2CCN1CC2 19608,C(=O)(CN1C(=O)CSc2ccccc21)N1CC(NC(C2C(C)CCC2)=O)(CO)C1 19609,c1(SCC2CC(N(C(C=C)C3CC3)C)C2)cccc(OCC(=O)OC)c1 19610,N1(C(C2(CNC(=O)CCc3cnco3)CC3(CC3)C2)=O)CCC(CO)C(O)C1 19611,O=C1CCC(C(N2CCN(C(=O)Cc3cn(C4CC4)cn3)C(CO)C2)=O)CCO1 19612,c1(CC)cc(Sc2oncc2C(N)=O)nc(Cc2cn(CC)nn2)n1 19613,C1(NC(CC)=O)(CCC(c2ccc(C(C)(C)C)cc2)O)CCOCC1 19614,c1(C(N(CCC)CCNC(=O)CC2CCCNC2=O)=O)ccc(C2CC2)nn1 19615,C#CC12CCC(C(N3CCC4(CC3)CC4CNC(=O)C(O)C(C)C)=O)(CC1)CC2 19616,C1(N(C(=O)CCOC(C)C)CC)CCCN(C(c2cc(C)[nH]n2)=O)C1 19617,c1(NC(C(C)NC(C(C)OC)=O)=O)cnc(F)nc1 19618,C1(CNC(C(C)C(F)F)=O)C(O)C(O)CN1C(=O)CC1(O)CCOCC1 19619,C1(N(C)C(c2cc(-c3cccnc3)no2)=O)CCC(NC(C2CC2(Cl)Cl)=O)CC1 19620,N#Cc1ccc(C=CC(=O)NCCNC(=O)Cc2csc3ccccc23)cc1 19621,c1(C(=O)NC2CC(C)(O)C2)ccc(N2CCNC2=O)c(F)c1 19622,CC1(F)CC2(CN(C(C3CCN(C(=O)C(C)(C)N=[N+]=[N-])CC3)=O)C2)C1 19623,c1(C(=O)NCC(N(C(=O)C=CC2CCCC2)C)C2CC2)cc2cccn2c(O)n1 19624,N1(C(c2cc(C)sc2)=O)CCC(CNC(=O)CCOCC(C)C)CC1C 19625,N1(C(c2scc(C)c2C)=O)CCC2(CC2NC(C2CC(C(C)C)=NO2)=O)C1 19626,C1(NC(CCCCCSC)=O)CCN(C(=O)CC2C=CS(=O)(=O)C2)CCC1(F)F 19627,C1(CCNC(C23CC(C)(C2)C3)=O)CCCCN1C(=O)C(C1(O)CCCC1)F 19628,CN1C(=O)CC(C(=O)NCC#N)C1Sc1ccccc1 19629,Cc1c(Br)cc(C(N2CC3CC3(C(=O)NCc3ccc[nH]3)C2)=O)cc1Br 19630,C(=O)(C(O)CC(N)=O)N1CC(N(C(=O)CNC(=O)NC2CCCCC2)C)C(O)C1 19631,c1(NC2(CC(=O)NC(CC(C)C)CO)CCC2)ncnc2c(Br)csc12 19632,N#CC1(C(=O)NC2CC(NC(=O)CCF)C2)CCCC(=O)C1 19633,C1(NC(=O)CC2CCCC2)CC12CCC(NC(c1ccc(Cl)cn1)=O)CC2 19634,N#Cc1ccccc1-n1cc(CNC(C2CC=CCC2)C(=O)O)cn1 19635,N1(C(c2c(CC)nccn2)=O)CCN(C)C(CNC(C2CCCCCC2)=O)C1 19636,CC1CN(C(C2(C)CCCN2C)=O)CCC1C(N1CCCC(C(N)=O)C1)=O 19637,CCCCC(CC)CC(=O)N(C)CC1(NC(C2Oc3ccccc3C2C)=O)CC1 19638,C1(C(N2C(C)CCC(C(N)=O)C2)=O)CCCCCCN1C(c1ccns1)=O 19639,c1(NC(c2cc(CNC(Cn3c(C)ccn3)=O)nn2C)=O)cccc(F)c1O 19640,C1(CNC(c2cn(CC)nc2)=O)COCCN1C(C1CC(F)CN1C)=O 19641,C(=O)(C(CCSC)NC(=O)C(CCC)OCC)NCC#CCC 19642,c1(C(N(C2CCN(C(=O)C=Cc3cccs3)C2)C)=O)cc(C(F)(F)F)ccn1 19643,N1(C(CC(=O)NCC2CC2)=O)CC2CCC1C(CNC(=O)CSC(F)(F)F)C2 19644,C1(C)(CNC(c2n(C)ncc2)=O)CCCN1C(=O)CCc1ccc(CO)cc1 19645,Cc1ccnc(C(=O)N(C2(C)CCN(c3nnnn3C)C2)Cc2ccccc2)n1 19646,c1(OC)sc(C(=O)NCC2(F)CN(C(=O)C(C)(Cl)Cl)C2)cc1Br 19647,C1(C(N(CC(CNC(C(C)=C(C)C)=O)(C)C)C)=O)CCCCC(F)(F)C1 19648,CC1C(NC(=O)CCC2CC2(F)F)CCCN1C(c1ccc(O)c(F)c1)=O 19649,c1(OC)cccc(F)c1C(=O)NC1CCN(C(C2CCC(F)CC2)=O)C1 19650,N1(C(C(c2cn(C)nc2)=O)=O)CCCC2(NC(=O)COC3CCCC3)CCCC12 19651,Cc1c(C(=O)NC23CC(NC(c4cc(O)ccc4F)=O)(C2)C3)cncc1Br 19652,C(CC)(CCC1CCC1)(c1n(C2(C(=O)NCC3CC4CCC3O4)CCC2)nnn1)OC 19653,c1(N2C(CNC(C3(C(=O)NC)CC3)=O)CC3COCC32)ncc2scc(Br)c2n1 19654,CC1CC(C(N2CCCC(CF)C2)=O)CCN1C(=O)CCc1cnccn1 19655,c1(CCC)ncc(C(=O)NCC2CCN(C(=O)C(C)c3ccsc3)C2)s1 19656,N1(c2nnc(C)c(C)n2)CC(C)(C)CCC1CNC(=O)C(C)C(C)C 19657,C1(C(=O)NC(C)Cc2ccnn2C)CC(O)CCN1C(=O)COC1(C)CCC1 19658,C#CCC(CC(=O)N1CCC=CC1COC)NC(C1CC(F)(F)C1(C)C)=O 19659,C1(C(C2CCC2)NC(=O)CC2CCCCO2)CCCCC1 19660,c1(C(=O)NC2C3(CC(NC(C(CC=C)(F)F)=O)C3)C2)ccc2cnc(C)n2c1 19661,N1(C(C2(OC)CCSC2)=O)CCOC(CCCNC(=O)COc2cnn(C)c2)C1 19662,c1(NCc2c(C)cc(C)cc2C)nc(C)cc(=NCc2ncccc2C(F)F)[nH]1 19663,c1(C(N2CCC(OCc3ccccn3)CC2)=O)cnccc1Cl 19664,c1(CC(N2CC=C(CNC(C3(CC4CC4)CC3)=O)CC2)=O)ccc2[nH]ccc2c1 19665,CC(C)(C)C(O)C(=O)NCC1CC(NC(c2cccc(-c3cnco3)c2)=O)C1 19666,C(CC(C(=O)O)NC(=O)CCc1cncnc1)c1cn(C(COC)COC)nn1 19667,CCCCS(=O)(=O)CC(=O)N1CC2C(CN=c3[nH]ncs3)C2C1 19668,C1(NC(=O)C=C2CCCCC2)CC2C1CCN2C(c1c[nH]c(C(F)(F)F)c1)=O 19669,N1(C(C=C(C)C2CC2)=O)CCSCC1C(=O)NC(C)C(N)=O 19670,c1(C2(C(NC(C(=O)NCCN(CC)CC)=Cc3cccs3)=O)CC2)ncccc1F 19671,C1(CNC(=O)OC(C)(C)C)(COC(C2C=CCCC2)=O)CC2(CC(F)C2)C1 19672,Cc1cc(C(N2CC(O)(CNC(=O)CC3(O)CCCN(C)C3)C2)=O)cc(C)c1F 19673,c1(-c2c(CC(=O)N(CCOC)Cc3ccccc3)scc2)ccc(C)c(C)c1F 19674,CCC(CC)OCC(=O)NCCC(C)NC(=O)CSC(F)F 19675,c1(OC)ccc(CNC(=O)C(c2ccc(I)s2)N(C2CCOC2)C(C)C)cc1 19676,C1(CCC(=O)N(CC(O)CNC(c2csc(C3CC3)n2)=O)C)CCC(C(N)=O)O1 19677,C1(C(=O)NCC(C)(C)F)C2CC(O)C(C2)N1C(c1cccc2[nH]ncc12)=O 19678,C1(C)(CNC(N(C(CS(CC)(=O)=O)C)C)=O)CCCCC1(F)F 19679,CC1(CCNC(C2(C)C=CCC2)=O)CCN(C(c2csc(Br)n2)=O)C1 19680,C(=O)(C1=CCOCC1)NC1CCC(NC(C2C(C#C)C2(C)C)=O)CC1 19681,CN1CC(C(=O)NCC2(NC(C3CC3c3cccs3)=O)CC2)NC1=O 19682,N1(C(C2(COC)CCCCC2)=O)CCN(C(=O)C(F)C(F)(F)F)C(C)C1 19683,C=CC(C)(C)CC(=O)NCC1(C)CCCN1C(=O)C=Cc1scnc1C 19684,CN(CCCC(=O)N1CCN(C)CC1CNC(=O)CC1CC(O)C1(C)C)N=O 19685,c1(C(=O)NC2(C)CCN(C(C3(CCO)CC3)=O)C2)ccc(Br)cc1[N+](=O)[O-] 19686,c1(C(N2CC(NC(C(C)N(CC)CC)=O)C2)=O)cc(OC)c2c(c1)CC(C)O2 19687,c1(C(=O)NCCCCCN(C(CNC(CC)=O)=O)C)ccc(N(C)C)cn1 19688,N1(C(CCCC#CC)=O)CC(CNC(=O)C(O)CC(C)C)CC(C)(C)C1 19689,N1(C(CSC2C(=O)OCC2)=O)CCC2(C1)CN(C(c1c(Cl)nsc1Cl)=O)C2 19690,N1(C(CC2C(C(=O)OC)C2(C)C)=O)CCC(NC(c2nn(C)cc2C)=O)C(C)C1 19691,c1(C(N(CCOCCNC(C2C(OC)CC2)=O)C)=O)csc2nccn12 19692,c1(C(=O)NCC(C)NC(c2n(CC)nc(C)c2)=O)ccc(F)c(C)c1C#N 19693,N1(C(c2occ(C)c2)=O)CC(C)(C)CC1C(=O)NCc1ccc(Cl)o1 19694,CC1=NOC(C)(C(=O)NCC(CO)NC(C2CCN(C)C2=O)=O)C1 19695,c1(C(N2C(CNC(c3ccc(C#C)cn3)=O)CCC2)=O)noc2c1CCCCC2 19696,C=CCC(C(=O)N(CC(C)O)CCNC(C12CCC(OC)(CC1)C2)=O)C(C)(C)C 19697,CCC(CC(=O)NC1CC(CNC(c2cc(Cl)c(F)cc2F)=O)C1)C(C)C 19698,N1(C(C(C(C)C)OC)=O)CC2C(NC(=O)CC(C)(C)C(C)(F)F)CS(=O)(=O)C2C1 19699,C1(NC(c2ccc(CNC(C(COC)COC)=O)cn2)=O)CN2CCC1(F)CC2 19700,Cn1nc(C(N2CCC(NC(C3CCN(CC(F)(F)F)C3)=O)C2)=O)cc1F 19701,C(=O)(C(F)C1=CCCCC1)NCc1ccc(CNC(C2C(=C)CC2)=O)c(F)c1 19702,C(=O)(CCC(F)(F)F)N1CCC(N(CCC)C(c2nn(CC)cc2Cl)=O)CC1 19703,c1(C(N(C)CC2(CNC(C3CC3Cl)=O)CC2)=O)ccc(CN2CCCCC2)o1 19704,c1(CS(N2CC(C(=O)OCC)C3(C2)CC3)(=O)=O)c[nH]c2nccc-2c1 19705,N1(C(C(C)(C)CCl)=O)CC2(CCN(C(c3cccc4nscc34)=O)C2)C1 19706,C(=O)(C1=CNC2=NCCCN12)NCC1N(C(CC2C(OCC)COCC2)=O)CC1 19707,c1(C(=O)NCC2C(NC(c3n(CCC)ccc3)=O)C2)cc2ccccn2n1 19708,c1(C(N2CC(C(C)NC(=O)C(C)C(F)F)C2)=O)ccc(N)c(F)c1F 19709,c1(C(N(C2CCCCN(C(C=CC(=O)N(C)C)=O)C2)C)=O)ccnc2c1CCC2 19710,c1(C(=O)NCCC(C(=O)NCC(CC)C#N)(C)C)nccc2[nH]ccc12 19711,C1(NC(CC(=O)OCC)=O)CN(C(c2ccnn2CC)=O)CC12CC2 19712,N1(C(c2c(C)scn2)=O)CCCC(N(C(=O)Cc2cc(Cl)cs2)C)CC1 19713,n1(CC)ccc(C(=O)N(CC(C)(C)NC(c2cc(C)c(Cl)s2)=O)C)cc1=O 19714,N1(C(c2scc(C)c2C)=O)CCN(C(C2CC(OC(F)(F)F)C2)=O)C(CCO)C1 19715,N1(C(C(C)NC(C=C)=O)=O)Cc2nccnc2CC1C(=O)NCC1CCOC1=O 19716,C1(NC(COC(c2cn(CCC)nc2)=O)=O)CN(C(=O)NC(C)(C)C)CC1C 19717,CC(N=c1ccc(C#N)n[nH]1)C1CCN(C(C2CCc3nn[nH]c3C2)=O)C1 19718,C1(NC(CN(S(CC)(=O)=O)C)=O)CCCCC1NC(=O)C=Cc1ncco1 19719,Cc1cccc(CC(=O)NC2CCCC(CNC(=O)CC(C)O)C2)c1 19720,c1(C(=O)NCC(CO)NC(C(C(C)C)OCC)=O)nc(C)c(C)nc1C 19721,CCC(CC(C)C)C(C(=O)Nc1c(C)cccc1C)N1CCCC(N2CCC2)C1 19722,c1(C(=O)NC(COC)CNC(C2CC(=O)N(C)C2)=O)ncc(Cl)cc1O 19723,N1(C(c2ccc(C)nc2C)=O)CC(NC(=O)CN2CC(=O)NC2=O)C(C2CC2)C1 19724,C1(C)(C(=O)NCCOCCN(C)C(c2cc(Br)cn2C)=O)CCCNC1=O 19725,N1(C(Cc2cn(CC)nn2)=O)CC(NC(=O)CNC=O)CC(F)(F)C1 19726,C(CCCCC(=O)NC(C)CCN(C(=O)Cc1cc(C2CC2)no1)C)OCC 19727,N1(C(C2C(OCC)C2)=O)CCC(NC(=O)C(N2CCCCCC2)C)C(C)C1 19728,C#Cc1ccc(C(=O)N(C)CC2(C(=O)NC3CC3(C)C)CC2)c(F)c1Cl.C(C)(=O)O 19729,c1(C(CNC(C(=O)NC2C(OC)CCC2)=O)OC)ccncc1F 19730,N1(C(C(C)N(C(CSC(C)C)=O)C)=O)CCCC(C)(O)C1 19731,C12(CNC(CCN(CCC)C)=O)CN(C(=O)CC=C(C)C)CC1CCO2 19732,c1(C(=O)NC(CCNC(c2nc(C)nn2C)=O)(C)C)nccc(N)c1Cl 19733,CC1CC(C(=O)NCC23CC(CNC(C4CC5CC5C4)=O)(CO2)C3)CC(C)C1 19734,c1(OC)cc(Br)c(C(=O)NCCN(C)C(c2nccc(C)c2N)=O)cc1OC 19735,N1(C(c2cc(C(=O)OC)oc2C)=O)CCC(n2cc(CO)nn2)C(O)C1 19736,c1(C(=O)NCC(CN(C(c2nc(C(C)=O)sc2)=O)C)C)nnc(C)cc1O 19737,Cc1noc(C)c1S(=O)(=O)N1CC2CN(S(=O)(=O)CCBr)C2C1 19738,c1(OC)cc(C(=O)NCC2CN(C(C3(OC)CC3)=O)C2)cc2cn(C)nc12 19739,c1(NC(=O)NCc2n(-c3c(C)cccc3C)nnn2)c(C)ccc(F)c1[N+](=O)[O-] 19740,C(=O)(N=c1ccn(CCC2CC2)[nH]1)C12CC(CNC(Cn3nnc(C)n3)=O)(C1)C2 19741,c1(C(=O)NCC2(O)CCCN(C(C3ON=C(CC)C3)=O)C2)cccn2nccc12 19742,N1(CC(=O)NCCC)CCS(=O)(=O)C(CCNNC(=O)CC2NC(=O)NC2=O)C1 19743,CCS(=O)(=O)CCC(C(=O)N1CC2CCC1C(CSC)C2)NC(=O)OC(C)(C)C 19744,N1(C(C(CC)CC2CCCCC2)=O)CC(C)CN(C(=O)Cn2cccn2)CC1C 19745,N1(C(C(C=C)C)=O)CC(O)(C2(CNC(=O)COCc3cccc(C)c3)CC2)C1 19746,c1(CCC)nc(=NC(C)CN(C(=O)Cn2cc3ncccc3n2)C)s[nH]1 19747,N1(C(c2c(CC)cno2)=O)CCC2C(C(=O)NCCCCC3CC3)C2C1 19748,c1(C(=O)NCC2(O)CCN(C(C3(C)CC3F)=O)CC2)coc2ccc(O)cc12 19749,C1(N(C)C)CN(C(C2CC2(Cl)Cl)=O)CC1CNC(c1csc(O)n1)=O 19750,c1(C(N2C3CC(NC(CCC(C)(C)F)=O)CC2CC3)=O)cnnc2ccccc12 19751,c1(C(=O)OC)ccccc1SCC(N1CC(C)(NC(=O)CC2CCC(C)O2)C1)=O 19752,N=c1[nH]c(=NCC2CC23CCOCC3)[nH]c(=NCCCCCC(=O)NC2CC2)[nH]1 19753,c1(C(N2C(C(=O)OC)(COC)CCC2)=O)ncn2c1CCNCC2 19754,CCC(CN(C)C)CC(=O)NCC1(O)CN(C(=O)CCC(C)N(C)C)C1 19755,c1(OC)ccc(CN2CCC(C(=O)N3CCCO3)CC2)c(I)c1 19756,N1(C(C(CC)(C)OC)=O)CCN(C)C(CNC(C2CN3CCC2CC3)=O)C1 19757,C12(C(=O)NCC3N(C(C(C(C)C)(C)O)=O)CC3)CC=CCN1CCC2 19758,C1(NC(c2c(CC)csc2)=O)COCCN(C(c2cn(C(C)C)cc2C)=O)C1 19759,Cc1cc(CO)oc1C(=O)NCC1(F)CC(CNC(=O)CC2CC3CC3C2)C1 19760,C(C1CN(C(=O)Cc2cnn(C)c2C)CC1C(=O)NCCCN1CC=CC1)=CC 19761,C1(NC(CC2CCN(C)C2=O)=O)CC2(C1)CC(NC(c1ccc(CO)cn1)=O)C2 19762,C1(C(N2CCN(C(c3c(CC)ncs3)=O)CC2COC)=O)CCc2nn[nH]c2C1 19763,C(C)(C(=O)NOOC)(N(C(C1CCC(Cc2cccc(C)n2)C1)=O)C)C1CC1 19764,c1(SC)nccnc1C(=O)NCC(C)N(C)C(C1CCC1(F)F)=O 19765,C1(C(c2nnnn2C)NCc2c(F)ccc(OC)c2)CCOC2(CCC2)C1 19766,Cc1cc(F)cc(C(=O)NCC2CN(C(C3CC4(CC4)CO3)=O)CC2(C)C)c1N 19767,n12c(C)cc(c1C)C=CC(=O)NC1CC1NC(=O)C2.C(=O)(C(C)CC)N.CCC 19768,N1(C(c2c(C)nn[nH]2)=O)CCCCCCC1C(N1CCC(C)(CO)C1)=O 19769,Cc1cn(C)nc1C(N1CCCC1CNC(C1(C)CNC(=O)N1)=O)=O 19770,C(=O)(C1=CCN(C(=O)CC(C)C2CC2)C1)N(C(CC(CC)C)C)C 19771,N1(C(C(CC)NC(C)=O)=O)CCn2cc(C(=O)Nc3cc(F)ccn3)nc2C1 19772,C1(C(=O)NC23CN(C(c4c(C)n(C)nn4)=O)C(CC2)C3)CNC(=O)CC12CCC2 19773,C#CCC(CC#C)C(=O)N1CC2CCN(C(=O)CCC(C)CC)C2C1 19774,C(=O)(C1CCCc2nncn21)NCCNC(c1c(C(F)F)ccc(C)c1)=O 19775,N1(C(CSCc2ccc(C(C)C)cc2)=O)CC2CC1CCC2NC(C1(C)CC1)=O 19776,c1(C(=O)NC2CC(C)(NC(C(CC)COC)=O)C2)cc(O)cc(F)c1 19777,N1(C(C(C)=C2CCC2)=O)CCC(C)(NC(c2ccncc2C)=O)CC1 19778,C1(CNC(C=CC=CC)=O)CN(C(c2n[nH]cc2C2CCC2)=O)CCC12CCC2 19779,C1(C(N(C2C(C)CC2)C)=O)CCC2CCC1N2C(c1cnn(C)c1Cl)=O 19780,N#CC1(C(=O)NC2CC(CNC(C3(S(N)(=O)=O)CCC3)=O)C2)CC2CC2C1 19781,C=CC(C)(O)CC(=O)N(C(CC(F)F)C(=O)NCC(C)Cc1cn[nH]c1)CC 19782,CCC(CC1CCCCC1)C(=O)NC1CCCCC1CNC(c1[nH]ccc1C)=O 19783,N1(C(C2(CC)CC2)=O)CCCC(C)(CNC(=O)CS(=O)(=O)NC2CC2)C1 19784,CC(C)C(C)(C)C(=O)NCc1nc(C(=O)NC2CNC(=O)C2)co1 19785,C1(C(=O)OC)Cc2ccccc2C1NC(=O)CC1C(=O)ON=C1C 19786,C1(F)(C(N(C)CC2C(C)C2)=O)CCN(C(C2CC(C)(C)CCO2)=O)CC1 19787,C12(CC)CN(C(=O)C(O)C(C)C)C(CNC(C3COCCN3C)=O)(C1)C2 19788,Cc1cccc(C(=O)N(CC(C)N(C(=O)CCSc2ccccc2)C)C)c1C 19789,Cn1c(CN(C=O)CCc2ccco2)ccc1C=O 19790,c1(C(=O)NC2CCC(NC(c3coc(O)n3)=O)CC2)ccc2c(c1)CCCC2=O 19791,C1(CC)CN(C(C2(C(N)=O)CC2)=O)CCC1NC(=O)CC12COCC(C1)C2 19792,C1(CNC(CCN(C(=O)CC2CCCC(O)C2)C)=O)OCCC1(C)C 19793,C(CCCCC(=O)N(C1CCN(C(c2cc(C)cs2)=O)C1)C)OCC 19794,c1(C(N(CC(=O)Nc2ccc(SC)nc2)CC#C)=O)[nH]ccc(=O)c1C 19795,C1(CN(C(c2ccc(OC)nn2)=O)C)CC2CCC1CC2 19796,C(CCN=C(NCc1cnc(C)cn1)NCc1cc(F)cnc1Cl)OC 19797,c1(C(C)NC(=O)NCc2cccc(NC(=O)OC(C)(C)C)c2)cccc(Br)c1F 19798,c1(OCC)ncc(C(=O)OCc2ccon2)cc1-c1cccc(C(C)O)c1 19799,C1(C(NOCCC#C)=O)CCC(C)(C)N(C(=O)C=CC2CCCN2C)C1 19800,C(=O)(CC(C)(C)NC(=O)C=CC1CCOC1)NC1C(CN(C)C)C1 19801,C1(C)(CNC(c2ccc(C(C)C)o2)=O)CN(C(=O)COC2(C)CCC2)CCO1 19802,n1(CC(=O)N(CCC(=O)NC2CCN(C(C)C)C2)C(C)C)ncn(C)c1=O 19803,N1(C(C2(CCC)CCC2)=O)CC2(CCC(CNC(=O)C(C)CC(C)(F)F)O2)C1 19804,Cc1cc(-n2cc(C(C(C)C)NC(=O)C(CO)NC(N)=O)nn2)cc(C)c1 19805,c1(NC(c2ncc(C)o2)C)nccc(=NC2COc3ccc(Br)cc32)[nH]1 19806,C1(CNC(c2nnc(CC)s2)=O)CC2COCC2N1C(c1sncc1C)=O 19807,N1(C(c2ccc(CC)s2)=O)CCC(NC(c2c(C(F)F)nn(C)c2C)=O)C(C)C1 19808,C1(CCC(=O)Nc2cccc(CC)c2)CCCCN(C(c2cccnc2C)=O)C1 19809,C(CNC(=O)COCC1CCC1)(CC(F)(F)F)NC(C(c1c(C)cncc1)C)=O 19810,C1(C(=O)NCC2(CO)CC2C(F)(F)F)CCCN(S(=O)(=O)C(F)(F)F)C1 19811,N1(C(CC(=C=C)C)=O)CC(CNC(=O)Cc2cnc[nH]2)CC(C)C1 19812,C1(NC(c2ccncc2Cl)=O)CC2CN(C(C3CCCSC3)=O)CC12 19813,C1(N(C)C(c2coc3c2COC3)=O)CCCC2CN(C(=O)CC3CC34CC4)CC12 19814,c1(C(N2CCC(O)(CNC(C3(C(=O)OCC)CC3)=O)C2)=O)cc(=O)cc(Cl)[nH]1 19815,N1(C(c2cc(C)c(Br)cn2)=O)CCC2C1CCCN2C(c1cc(O)nc(O)n1)=O 19816,c1(C(=O)NC(C(=O)NCCNC(=O)NC)CCOC)cccc2ccoc12 19817,C1(NC(C(C)C(C)(F)F)=O)CCOC2(CCN(C(C3CC4CC4C3)=O)CC2)C1 19818,C1(N(C(=O)C(C)n2cccn2)CC(=O)NCC)CCCC12CCNCC2.N(C)C 19819,c1(C(=O)NC(COC)CC(F)(F)F)ccc2n1CCNC2 19820,N1(C(c2nc(CNC(C3N(C)CCOC3)=O)oc2)=O)CCC(O)C(O)C1 19821,C1(CC(=O)N(C2CCN(C(C34COCC(C3)C4)=O)C2)CC)CC2CCC1C2 19822,Cc1cccc(F)c1CC(=O)NCc1ncoc1CNC(=O)CC1COCC1O 19823,c1(C(=O)NCC(CC)NC(C2CNC(=O)N2C)=O)ccc2ccc(O)nc2n1 19824,CC1CCCN(C(c2cccnn2)=O)C1CCNC(c1cc(F)ccc1Br)=O 19825,N1(C(C(C)OCC#C)=O)CCCC(C)(CNC(=O)CC2(C)CCCO2)C1 19826,N(C(=NCC=C1CCCC1)NC(c1ccccc1)C)CC(CC=C)(C)C 19827,c1(CC)nc(O)c(C(=O)NC2CCCCC2CNC(C2(C)CC=CC2)=O)cc1C 19828,N1(C(CC=CC)=O)CCN(C(=O)CSCCC)CC1CC 19829,C1(C(=O)NC2(C(C)O)CC2)CCCC(NC(C2COCC2(C)C)=O)C1 19830,N1(C(c2cc(I)c(F)cc2F)=O)CCC2C(CCN2Cc2cccc(Br)c2Cl)C1 19831,N1(C(Cn2c(CC)nnn2)=O)CCC2CCC(C1)N2Cc1cc(C(C)(C)C)on1 19832,C(C(C)C(F)C(=O)NCc1csc(C)c1C)NC(c1ncn(CC)c1)=O 19833,CC1C(C(=O)NC23CC(NC(C4OC(C)(C)OC4(C)C)=O)(C2)C3)C(O)C(=O)N1C 19834,c1(NC(C2CCCCN2C(c2ccnnc2O)=O)=O)cc(Cl)ccc1CO 19835,CCC1=C(C(=O)NCC(C)CNC(c2c(C)nn(C)c2C(F)(F)F)=O)SCCO1 19836,c1(NC(C2CN(C(C(COC(C)C)NC(C)=O)=O)C2)C)nccc(C)n1 19837,C1(C(=O)NCC(C)(C)NC(c2cc(C(F)(F)F)no2)=O)C2CC2C2CC12 19838,C1(CC(=O)NC2C(OC)CCCC2)C2CCCC2N1C(c1nscc1C)=O 19839,N1(C(CC2N(C(CSCCOC)=O)CCC2(C)C)=O)CCC2(C=CCO2)C1 19840,N1(C(c2ncc(C)cc2F)=O)CCC2C(CCCN2C(=O)CC(C)(F)F)C1 19841,C1(C(=O)NCCN(CCC)C(c2ccnn2CC(C)C)=O)CCCC1S(C)(=O)=O 19842,CCS(=O)CC(=O)NCC(c1ccc(F)cc1)NC(C1(OC)CC1)=O 19843,Cn1nc(C2CC2)cc1C(=O)NCCCCCCNC(=O)CC1CNC(=O)C1 19844,C(=O)(CC(C)N(C)C1CC1)NCC(C)NC(=O)CCc1sccc1Br 19845,N1(C(C(C(CC)C)O)=O)CCCC2(C1)CN(C(=O)CN1CCP(C)(=O)CC1)C2 19846,CC1(C)CCOC(CC(=O)NC2CN(C(=O)CSCC3CCCO3)CC2O)C1 19847,c1(C(=O)NCC(CC=C)NC(c2cscc2C)=O)cc(N(C)C)ccn1 19848,c1(-c2c(C)nc3scc(C)n32)nc(C2Cc3ccccc32)nn1C 19849,c1(NC(CNC(c2ccc(OC)nc2)=O)CC(C)C)c(Cl)cccc1[N+](=O)[O-] 19850,N#CC1(C(N2CC(CNC(=O)CCCCCNC(N)=O)C2)=O)CC2CCC1CC2 19851,C(=O)(C(CC(N)=O)NC(=O)COC1CCCOC1)NCC(C=C)O 19852,C=CCCCC(=O)NCCC1(C(=O)NC2(C3CCC3)CC2)CCC1 19853,CC(C(C)(C)CO)NC(=O)C(C)(C1CC1)N(C(=O)COc1ccsn1)C 19854,c1(C(=O)NCC2(C(F)F)CCN(C(C(CC)OCC)=O)C2)c(Cl)ccc(C)c1O 19855,N1(C(C2CCC(C)CC2)=O)CCC(NC(c2cnn(C3CC3)c2)=O)CC(C)(C)C1 19856,c1(NCCC(C)C)cc(S(=O)(=O)NC(Cc2ccc(Cl)cc2)CO)ccc1C#N 19857,N1(C(CCCC)=O)CCN(C2CCC(NC(C3(C)CCC(=O)N3)=O)CC2)CC1 19858,C1(NC(c2cn(C)nc2C2CC2)=O)CCCCN(C(=O)CO)CC1 19859,N1(C(C(CC)OCC)=O)CCc2nc(CNC(c3cn(C)nc3C)=O)sc2C1 19860,C(N=c1[nH]cnc2c1COC2)C1(CNC(C2CC3CCC2O3)=O)CCC1 19861,C(=O)(C(CC)NC(C)=O)N(CCNC(C1CCCN1C(=O)C(F)(F)F)=O)CC 19862,C(CCCCCC(=O)NCCC1CCC(=O)N1)NC(C(=Cc1cn[nH]c1)C)=O 19863,C12(CNC(c3c(C)coc3C3CC3)=O)CCCC1CCN2C(c1cc[nH]c1)=O 19864,N1(C(Cc2cc(C)sc2)=O)CC2(CO)CC1(C(=O)NC1CC(O)CC1O)C2 19865,C(=O)(C(C(C)CC)N(C(=O)CCN1CCCCC1)C)N(CC#C)CCF 19866,C1(NC(=O)CCF)CN(C(=O)Cc2nnc(-c3ccncc3)o2)CC1C1CC1 19867,c1(CNC(C2N(C(C)C)CCC2)=O)ccc(CNC(C2CC2(C)C)=O)cc1F 19868,N1(C(C2N(C)C(=O)CC2)=O)CCC(O)(C2CCN(C(=O)C3=CCC3)CC2)CC1 19869,N1(C(CSCCCC)=O)CCC2(CC1)CCN(C(C1CCC3CC3C1)=O)C2 19870,N1(C(C2(C(N)=O)CC2)=O)CC(NC(=O)CS(=O)(=O)CCO)C(C2CC2)C1 19871,c1(CNC(C2CC2CF)=O)ccccc1CO.C12(CCC1)CC(=O)NCC2 19872,c1(C(=O)NCC2CC(NC(c3nocc3Cl)=O)C2)c[nH]c2ccc(Cl)cc2c1=O 19873,c1(C(=O)OC)ccc(N2CC(CCNC(=O)C(c3ccnn3C)C)(OC)C2)nc1 19874,c1(NC(C2CCCC2NC(c2cn(-c3ccccc3)nn2)=O)=O)c[nH]nc1Br 19875,c1(C(=O)NC(C2CN(C(c3conc3C(F)(F)F)=O)C2)C)ccncc1C(F)F 19876,Cc1ccncc1CC(=O)NCC(C)(C)NC(c1cnc(N2CCOCC2)s1)=O 19877,c1(C(=O)NC2C=CC(C(=O)NC(c3ncc[nH]3)CC)C2)ccnc(C)c1C 19878,Cc1cccc(-c2cncc(C(=O)NCC(O)CCNC(C3CCCS3)=O)c2)c1 19879,CCCC(O)CC(=O)NCC1(NC(=O)CCNC(=O)C(C)(C)C)CCC1 19880,CC(C)(C)C1=NOC(C(N2CC3CC3(NC(c3ccns3)=O)C2)=O)C1 19881,C1(NC(C(=O)NCC)=O)C2CCCN(Cc3cc(C)ns3)C2C1(C)C 19882,c1(C(N2CC(O)(CCNC(C3C(C)(C(F)F)C3)=O)C2)=O)cccc([N+](=O)[O-])c1N 19883,Cc1cc(C(C)NC(=O)NC(C)CCNc2[nH]nnc2C)cs1 19884,C1(CC)CN(C(c2cncn2C)=O)CCC1CNC(c1ccnn1C)=O 19885,C1(C(=O)NCc2n(C)ccn2)CC(F)CN(C(c2cc(O)ccc2O)=O)C1 19886,N1(C(C(CC(C)C)(F)F)=O)CCCC2(C1)CN(C(c1ccnn(C)c1=O)=O)C2 19887,C(=O)(CS(=O)(=O)NC1CC1)NCC(C)CNC(=O)C(N1CCCC1)C1CC1 19888,c1(C(N2C(C)CN(C(C3(C)CC3(F)F)=O)CC2)=O)cccn2ccnc12 19889,N1(CC)CC(C(=O)NC2CN(C(C3(F)CCCC3)=O)CC2C)CC1=O 19890,c1(C(=O)NCC2CC(NC(=O)C(F)(F)c3nccs3)C2)cc2c(Cl)cncc2s1 19891,c1(C(N(CCCNC(C(CCC)NC(C)=O)=O)CC)=O)c(Cl)ccc(Cl)c1O 19892,C12(CNC(C(C)(C)SC)=O)CCC(CN(C(C34CCC(C)(C3)OC4)=O)C1)C2 19893,C1(CNC(CCN(C)CC)=O)C(C2CC2)CCN1C(=O)C#CC1(C)CC1 19894,Cc1cccc(Cl)c1C(N1CC(CC(N2CCC(CF)CC2)=O)C1)=O 19895,c1(C(=O)NC2CCC(C)N(C(C3C4CC5C(C4)C35)=O)C2)ccc2nnn(O)c2c1 19896,CC(C)CC(C(=O)NC1CCCCC1CCO)ONC(=O)CC1(C)CCOC1 19897,N1(C(C(=O)NCC=C)c2cccs2)CCc2ncncc2C1 19898,C1(C(=O)NCC2CCCN(C(c3cnc(C)[nH]3)=O)C2)COC2(CCC2)C1 19899,c1(NC(C)=O)ccc(NC(=O)CC2CCCN(C(=O)CCCCC#N)C2)cc1C 19900,c1(C(=O)OC)ccc(COC(c2occc2Br)=O)c(OC)c1 19901,C(=O)(C(CC(C)C)N(C(=O)Cc1ccccc1C)C)N1CC(C(N)=O)(OC)C1 19902,c1(C(C)=O)ccc(C(=O)NCC2CC(C)N(C(=O)OC(C)(C)C)C2)cc1Cl 19903,Cc1ncc([N+](=O)[O-])n1CC(=O)NC1CC(CCNC(C2CC(C)CCO2)=O)C1 19904,C12(CNC(C(CC(C)C)N(C)C)=O)CN(C(c3cc(Cl)no3)=O)CC1CCO2 19905,Cc1sc(C(=O)NCC(CO)NC(c2ncccn2)=O)cc1-c1ccc(F)cc1 19906,c1(-n2c(C)nnn2)c(F)cc(C(=O)N(C)CCc2ccccc2F)cc1F 19907,C1(C(=O)NCC(=O)N(CC)CC)CCC(C(C)C)N1C(c1cc(CO)c(C)o1)=O 19908,C1(CC)CCN(C(=O)CCN(CC)CC2CC2)C1.C1(C)(C)CNC(=O)CO1 19909,c1(CC(N2CC(O)(C(C)NC(C=C(C)C3CC3)=O)C2)=O)cc(F)ccc1F 19910,C1(CNC(c2ccc(F)cc2)=O)CCC2(CN(C(C3(CO)CCC3)=O)C2)O1 19911,C1(SC)CN(C(=O)CC(F)(F)F)CC1C(=O)NC1CC(N(C)C)C1 19912,O=C(C1=CS(=O)CCC1)N1CCN(C(c2ccccn2)=O)C(CC2CC2)C1 19913,c1(C(=O)NC(CC2CN(C(C3(CC#C)CC3)=O)C2)C)ccn(CC)c(=O)c1 19914,c1(C(=O)NCC2CN(C(c3n(C(C)C)ccc3)=O)C2)cc2n(c1)CCC2 19915,c1(C(=O)NC2(C)CCN(C(=O)CC3CCCC(=O)C3)C2)onc2c1CCCC2 19916,N1(C(Cc2n(C)c(S)nn2)=O)CCCC(F)(CNC(=O)CC2CNC(=O)O2)C1 19917,Cc1ccn(CC(=O)NC2CC(N(C)C(c3coc(C4CC4)n3)=O)C2)c(=O)c1 19918,c1(C(N2C3C(NC(c4ccc(C)nn4)=O)C(C3)C2)=O)n[nH]cc1[N+](=O)[O-] 19919,C1(CC)CC(O)CN1C(=O)C(CC1CCC1)NC(=O)C=CC(=O)OC(C)(C)C 19920,N1(C(c2c(C)cc(N)cn2)=O)CCCC2(CCCCC2NC(c2cn[nH]c2)=O)C1 19921,N1(C(C2C(OC)C2)=O)CC(NC(c2nccc3[nH]ccc23)=O)C2(CCOCC2)C1 19922,CCC(CCOC)C(=O)NCC1CC(OC)CN1C(c1ccccc1CC#N)=O 19923,S(=O)(=O)(CC(=O)NC1CCC(NC(c2ccnn2C2CCCC2)=O)C1)NC 19924,C=CCCCCC(=O)NC(CO)C(C)NC(c1ccnc(OCCOC)c1)=O 19925,N1(C(C2CCC2)=O)CC2C3CCC(C2C1)N(C(c1c(F)cc(F)cc1Cl)=O)C3 19926,CON1CCC(CN(C)Cc2ccc(O)cc2)CC1 19927,N1(C(c2c(CC)ocn2)=O)CCC(NC(C23CCC(C2)C3(C)C)=O)C(C(N)=O)C1 19928,c1(C(N2CC(NC(=O)C=C(Cl)Cl)C(CO)CC2)=O)ccn2nccc2n1 19929,c1(Oc2ccc(OC)cc2C=Cc2ccco2)cccc2sc(CO)nc12 19930,c1(C(=O)NCC2(NC(C(CCCC)O)=O)CCOC2)ccc2c(c1)NC(=O)C2=O 19931,c1(C(=O)NCC2CC(OC)CN2C(=O)C(C)NC(C)(C)C)ccc2ccsc2c1 19932,CC1(C)CC(NC(=O)C(=Cc2ccccc2)C#N)CN(C(c2coc(Br)c2)=O)C1 19933,c1(C(C)C)ccoc1C(=O)NCCCCNC(c1ccc(C2CCCO2)[nH]1)=O 19934,S(=O)(=O)(C=Cc1ccccc1)NC1C(F)(F)CCN(C(=O)CN2CCOCC2)C1 19935,N1(C(C(CSC)C)=O)CC(O)CC1CNC(c1nc(C2CC2)cs1)=O 19936,C12(C(=O)NCC3C(NC(CSCCOC)=O)CCCC3)CCN(CC1)S(=O)(=O)C2 19937,C1(CC)C(CC(=O)NCCN(C(=O)C(C)Sc2ccccc2)CC2CC2)C1(F)F 19938,N1(C(CC(CCC)O)=O)CC2(CCC2)CC1CNC(C1(NC(C)=O)CCCC1)=O 19939,c1(C(=O)NCC(CNC(CC2(OC)CCCCC2)=O)F)c(C)cc(F)cc1C 19940,N1(C(c2cccc(COC)n2)=O)CCC2CCN(C(c3ccoc3Cl)=O)CC12 19941,C1(NC(C2C(CC)OCC2)=O)CC=C(C(=O)NC(CC)C(=O)OC)C1 19942,CC(C(=O)NCC1CC2(C1)CN(C(=O)Cc1cccc(C#N)c1)C2)C(C)(F)F 19943,C1(C(=O)OCC)(OC)CCN(C(=O)C(n2cc(-c3csc(C4CC4)n3)nn2)C)C1 19944,O=C(CCC(F)F)NCCCCNC(C1(CC2CCCC2)CCCC1)=O 19945,C(=O)(CCC(N)=O)N(CCC(=O)NCC(O)(CO)OC)C 19946,C1(C(=O)NC2C=CC(CC(=O)NCC3CCCS3)C2)(OC)CCSC1 19947,c1(OC)ccc(C(n2cc(-c3cc(Cl)ccc3C)nn2)C)c(Br)c1 19948,c1(OC2CCCC(C(=O)NCCNC(CC(=C=C)C)=O)C2)ccccc1C#N 19949,C(C1CCCC1)=CC(=O)NC1CCC1CNC(C1CCC(C(F)(F)F)O1)=O 19950,C(=O)(C1=CCCCCC1)NC(C(N1CC[Si](C)(C)C1)=O)C1CCOC1 19951,c1(NC(COC(C(CCOC)C)=O)=O)ccc2c(c1)CCC2 19952,Cc1cc(C)n(C(C)CC(=O)NC(C2CCCN2C(=O)CCC(=O)C2CC2)C)n1 19953,C(=O)(C(C)CC(=O)c1ccccc1F)NCCNC(C(N1CCNC1=O)C)=O 19954,C1(O)(C(=O)NC(CN(C(CC2(C=C)CCCCC2)=O)C)(C)C)CN2CCC1CC2 19955,c1(OC)cc(C(=O)NCCCN(C(=O)C(C)C(F)F)Cc2ccccc2)ncn1 19956,c1(C(N2CC(CNC(C3CC(OC(F)F)C3)=O)C3(CC3)C2)=O)cccc(F)c1Cl 19957,c1(C(N2CC(O)CC(NC(c3cc(C#N)sc3)=O)C2)=O)cc2nc[nH]c2cn1 19958,Cc1sc(C(F)(F)F)c(C(=O)NC(CNC(=O)C(F)C(F)(F)F)CO)c1C 19959,C1(NC(c2c(C)cn(C)n2)=O)C2COCC1CN(C(=O)C=Cc1scnc1C)C2 19960,C(C)(C)(C(=O)NC(Cc1ccco1)C(=O)OC)N(CC)CC 19961,N1(C(CC=CCNC(C2(CCN=[N+]=[N-])CC2)=O)=O)CC2CCCCC2C1 19962,N1(C(C(CC)CC2CCCC2)=O)CCN(c2nc(C)cc(C)n2)C(C)C1 19963,O=C(C1=CC2(CCN(C(=O)C(F)n3ccnc3)C2)C1)NCC1(CC2CC2)CC1 19964,N1(C(=O)CC(F)F)CCN(C(c2ccc(C(F)(F)F)cn2)=O)C(CF)C1 19965,C(=O)(C(C)(C)C1=CCN(C(=O)CC=CCCCCC)C1)NCCCC=C 19966,N1(C(C(C2CC2)OC)=O)CCCC(N(C)C(c2cccc(F)c2SC)=O)CC1 19967,c1(C(=O)NCC(CC(C)C)NC(C(COC)(C)C)=O)cnn2cc(C)cnc12 19968,N1(C(c2c(CC)csc2)=O)CCCC(C)(C(N2CCC(CC(=O)OC)C2)=O)C1 19969,CC(CC(F)(F)F)C(=O)NCC(C)(C)CCNC(c1cccc(NCC#N)c1)=O 19970,c1(C(N2CC(OC)C(NC(=O)C=CC3CCCN3C)C2)=O)ccc2ocnc2n1 19971,C1(Oc2c(NC(N3CC(OC)C3)=O)cccc2)CCc2c[nH]nc2C1 19972,N1(C(Cc2c(C)ncs2)=O)CC2CC(N(C(=O)COCCOCCO)C)C1C2 19973,N1(C(C(F)=C(C)C)=O)CCN(C(C2CC2(Cl)Cl)=O)C(C(C)C)C1 19974,N1(C(CC(n2c(CC)ncc2)C)=O)CCCC2CN(C(=O)CC(C)OC)CC12 19975,Cc1nc(NCCc2csc(Br)c2)cc(=NC(C)c2nncs2)[nH]1 19976,C1(N(C)C(c2cncnc2)=O)CCCC2CN(C(=O)CC3(O)CCC3)CC12 19977,c1(C(N2CC(COC)N(C(=O)CCSCC(N)=O)CC2)=O)cc2oc(C)cc2[nH]1 19978,C(c1c(C)nn(C)c1Cl)=CC(=O)NCCN(C(c1cnc(S)[nH]1)=O)CC 19979,c1(C(=O)NCC=CC(=O)NCCC(C)NC(=O)N(C)C)cccn2c(O)nnc12 19980,N1(C(=O)N(CCO)Cc2cncnc2)CC(c2cccc(F)c2)C(c2ccccc2)C1 19981,Cn1cc[nH]c(=NNC(=O)NCC2C(C(=O)O)C2(C)C)c1=O 19982,C12(CNC(c3n(CC(C)C)ncc3)=O)CCCC1CNC2 19983,O=C1CCOCCN1Cc1cn(CC2CCN2C(=O)CCc2cc(Br)ccc2F)nn1 19984,C(CC(C)C(=O)NCC(CNC(=O)Cc1ccncc1Cl)CO)=CC 19985,C1(CCOC)(NC(c2ccc(Br)o2)=O)CCN(C(=O)Cc2ccco2)C1 19986,c1(C(N2CC3(CCN(C(C4(NC(C)C)CC4)=O)C3)C2)=O)cccc2ccn(C)c12 19987,n1(CC)cncc1CC(N1CC(c2ccccc2)(CO)C1)=O 19988,CC1(C)CC(NC(=O)Cc2ccc(Br)cn2)CN(C(C2COCCO2)=O)C1 19989,Cc1c(Cl)nc[nH]c1=NCC(O)CNC(C1CCCCC12CCC2)=O 19990,N1(C(C=CCC)=O)CC(C(=O)NOCC2CCCNC2=O)C(COCC)C1 19991,C(=O)(CC1=CCN(C)CC1)N1CCC(C)C1C(N1CC[Si](C)(C)CC1)=O 19992,c1(C(=O)NC2CC(CNC(CCNC(COC)=O)=O)C2)cc(C)n(C(C)C)n1 19993,c1(C(N(C(CN(C(C(COC)OC)=O)C)C)C)=O)ccc2ncccc2c1F 19994,O=C(CCC(F)(F)F)NCC1CC1NC(c1cnn[nH]1)=O 19995,c1(CNC(CC(C)CF)=O)nc(CNC(=O)C(C)c2ccco2)cc(O)n1 19996,C1(N(C(C2ON=C(CC)C2)=O)C)CCC2CN(C(c3cccc(F)c3N)=O)CC12 19997,C1(C(=O)NCC(C)(CNC(c2cc(C3CC3C)on2)=O)OC)CC2(CCC2)C1 19998,N1(C(=O)C=CC=C(Cl)Cl)CCC(F)(CNC(C2CC(C(F)(F)F)C2)=O)CC1 19999,c1(C(N2CCC3(NC(c4ccsc4)=O)C(CC2)C3)=O)cc2c(O)ncnc2cn1 20000,C(=O)(C(F)CCC(C)(C)C)N1CCC(CC#C)(C(=O)NCC2CC2(Cl)Cl)C1 20001,C1(C(=O)NC2(CO)CN(C(c3n(C)c(Cl)nc3)=O)C2)CC1C1CCCC1 20002,C#CCC(CC(F)F)C(=O)NC1(C)CCCN(C(C2CCC=CCCC2)=O)C1 20003,CCCC(CCC)C(=O)NC1CCN(C(c2c[nH]nc2Br)=O)CC1CC 20004,C(=O)(CN1C(=O)COc2ccccc21)NCCCc1cn(-c2ncc(C)s2)nn1 20005,C(c1cccc(F)c1)=C(C(N1C(CNC(C(N2CCCC(O)C2)C)=O)CC1)=O)F 20006,C1(N(C(=O)Cc2ccc(OCC#N)cc2)C)CN(C(=O)C(C)(C)F)CC1(C)C 20007,N1(C(C(C(C)C)C)=O)CCC2(CC2NC(c2ncccc2F)=O)C1 20008,C1(CC(C(C)CNC(=O)OC)=O)C(=O)NN=C1C.C1(C2C(=O)N2)CCCCC1 20009,C1(C(N(CCN(C)C)CCO)=O)CC2CCC1N2C(=O)CCCOC(C)(C)C 20010,C1(NC(C(C)n2cncn2)=O)CC2(CCCN(C(C3CC4CCC3C4)=O)C2)C1 20011,N1(C(C(C)(C)CCF)=O)CCC2CN(C(C3CC(=O)OC3(C)C)=O)C2C1 20012,C1(C(N2CCC(C)(NC(c3n(CC)ncn3)=O)CC2)=O)CCC2C(CC1)C2(F)F 20013,C(C(N=[N+]=[N-])C(=O)NCC(O)CNC(c1csc(C(C)C)n1)=O)OCC 20014,CC1(C)C(C)(C)C1(F)C(=O)NCCCNC(c1cccc(N)c1F)=O 20015,C(=O)(CC(C)(C)COC)NCCOC(c1nc(C(CC)CC)cs1)=O 20016,c1(N(CCCN=[N+]=[N-])CCOC)ccccc1C1CCC1 20017,c1(C(=O)NCC2N(C(C3CC(OC)C3)=O)CC(O)C2)cccc2c1CNC2=O 20018,CC1(CNC(=O)CC2CCCO2)CN(C(c2ccsc2C(F)(F)F)=O)CCO1 20019,CN=c1[nH]c(=NCC(C)F)[nH]c(=NC2CCCN(Cc3ccccc3)C2)[nH]1 20020,CC1(NC(=O)CC2(O)CCC2)CCC(NC(C2CS(=O)C2)=O)CC1 20021,c1(NCCN2C(CC(=O)OCC)CCCC2)ccc(C#N)cc1CC 20022,C1(NC(C(N)=O)=O)CC(C2CCN(C(c3n[nH]c4c3CCOC4)=O)CC2)C1 20023,C1(n2cc(C(C(OC)OCOC)C)nn2)CN(C(c2conc2C)=O)CC1C 20024,c1(C(N2CC(CC(C)NC(=O)CCS(C)(=O)=O)C2)=O)ccc2c(c1)OCO2 20025,N1(C(c2cc(CCC)[nH]n2)=O)CCC(O)C(NC(c2ncoc2CC)=O)C1 20026,c1(NC(C)=O)ccc(C(=O)NCCCN(C)C(c2ccc(CO)cn2)=O)cc1F 20027,C1(C(N2CCC(CO)C(O)CC2)=O)CC12CCN(C(C1(CO)CC1)=O)CC2 20028,N1(C(N(C)C)=O)CCC(C(=O)NCC(C2CCCC2)NC(=O)CC2(C)CC2)C1 20029,O=C(C1=COCCO1)NCC1(NC(C2CC3C=CC2C3)=O)CCCCC1 20030,CC(=O)C(C)CC(C)C(=O)NC(C(=O)NCCSCCCO)C1(O)CCC1 20031,c1(C(N(CCNC(c2c[nH]nc2Cl)=O)CC)=O)cc(OC)cc(C)c1 20032,C1(CC(NOC(CC)CC)=O)CC2(C1)CN(C(=O)COCCCOC)C2 20033,c1(-n2cc(C3C(=C)CC3)nn2)ccncc1Br 20034,c1(C(N(C2CCN(C(C(C(C)C)OC)=O)C2)C)=O)cc2nccn2c(O)n1 20035,C1(NC(CC(CC)C)=O)CCN(C(=O)CCN(CCCCOC)C)CC1F 20036,N1(C(C)=O)CC2(CC(S(=O)(=O)N3CC(N4CCOCC4)C3)C2)C1 20037,c1(C(=O)NC(COC)CNC(=O)C(C)(COC)OC(C)=O)cc2nc(C)sc2[nH]1 20038,N1(C(C2(C#N)CCC2)C(=O)NCC(F)F)CCN(Cc2ccc(F)cc2)CC1 20039,C(CCN=c1[nH]c(=NC2CCc3cccnc32)[nH]c2c1SCC2)=CC=C 20040,C(O)(C(=O)O)(C(F)(F)F)n1cc(Cc2oc(C)c(C(N3CC4CC3(CO)C4)=O)n2)nn1 20041,N1(C(COC)=O)CC2CCC2(CNC(=O)C(C2CCCCCC2)O)C1 20042,C1(C)(CNC(COc2ccc(C)cc2)=O)CN(C(=O)CCCCCF)C(C)(C)C1 20043,C(=O)(C1(C)CCc2ccccc21)N1C2C(CNC(C3C(C)C3)=O)C(C2)C1 20044,c1(C(=O)NCC2CN(C(C(CCC)C)=O)CC2(F)F)cnc2c(cnn2C)c1 20045,C1(NC(c2cc(SC)oc2C)=O)CN(C(C2(C)CCCCO2)=O)CCC1O 20046,N1(CC)CCCN(C(C2OCCC2NC(=O)C(C2CCCCC2)O)=O)CC1 20047,N1(C(c2cnc(OC)s2)=O)CCCC1C1CCCN1C(=O)C=Cc1nc(C)co1 20048,C(CCC(C)(C)NC(c1sc(C(C)OC)nc1C)=O)NC(C(CC1CC1)OC)=O 20049,C1(C(N2CC(OCC(=O)NC)C2)=O)CCC(O)CN1C(C12CC(C#N)(C1)C2)=O 20050,n1(CC(N2CCN(C(C(CCC)O)=O)C(C)C2)=O)cnc2ccccc12 20051,C(=O)(CC(C(=C)C)Oc1cnn(C)c1)N1CCC(C#C)C1 20052,CC1CN(C(c2ncccc2C(F)(F)F)=O)CC1(C)CNC(=O)Cn1cncn1 20053,CC1=C(C)CC(C(=O)NCCC(C)(C)CNC(C2CC3CC3C2)=O)CC1 20054,C1(NC(C(C)C#N)=O)CN(C(c2ccc(CN3CCOCC3)s2)=O)CC12CC2 20055,c1(C(N2CCC3(C(CNC(CC=C=C)=O)C3)CC2)=O)coc2c(OC)cccc12 20056,CC(C)CC(C)(CNC(=O)COC1CCN(C)CC1)NC(c1cnccc1Cl)=O 20057,CCCCC(C(=O)NCC1CCCCN1C)NC(=O)CN(C(=O)COC)C 20058,CC(C)CC(C)(CNC(c1ccc(C(N)=O)s1)=O)NC(c1ncc(F)cc1F)=O 20059,c1(CC)nnc2c(C(=O)NC3CCCC3NC(C3CCCN3CC)=O)cccn12 20060,C(CCCC(=O)NCCOc1ncccn1)N(C(=O)C=Cc1ccsc1)C 20061,C1(NC(C=CCC)=O)CN(C(c2cccc(N)c2O)=O)CCC1CO 20062,N1(C(C2N(C(C)=O)CCCC2)=O)CCC(C)C(N(C(=O)Cc2cnco2)C)C1 20063,c1(C(N2CCC(NC(CNC(=O)OC)=O)C(O)C2)=O)cc2c(C)[nH]nc2s1 20064,N1(C(c2c(C)cc[nH]2)=O)CCN(C(=O)C(C)Cc2cccc(F)c2)CC(C)(F)C1 20065,c1(N2CC(N3CCN(C(C)=O)CC3)C(C)C2)ccnc2cc(O)ccc12 20066,c1(C(N2CC(NC(CC(C=C)C)=O)C(C)C2)=O)cc(Cl)ncc1O 20067,C1(C(N2CCC(O)(CCNC(c3ccsn3)=O)C2)=O)CC2CC(C1)CS(=O)(=O)C2 20068,O=C(C(Cl)=CCl)NCC1CC(NC(c2csc(C(F)(F)F)n2)=O)C1 20069,c1(N(CC)CC)ccc(C(=O)NCCNC(=O)C(C)NC(C2CCC2)=O)cn1 20070,N1(C(c2cccc(C)c2)=O)CCN(C(=O)CC2CCC(C(F)(F)F)O2)CC1CO 20071,CC(=O)C(C)CC(C)C(=O)N1CCN(C(=O)C#CC2CCC2)C(C(C)C)C1 20072,N1(C(CCC(=C)C)=O)CCC(CNC(=O)CC2(COC)CC2)(OC)CC1 20073,C1(C)(C(N2CCCC(=C)C2)=O)CCN(C(c2cc(C)ccc2F)=O)CC1 20074,Cn1cc2c(n1)CC(CN1CCCC(C(c3ccccc3)O)C1)CC2 20075,N1(C(C2CC(OC)C2)=O)CCC(NC(=O)C=CC(F)(F)F)C1C(C)(C)C 20076,C(=O)(CCC(=O)N(C)C)N(C1CCN(C(CCCSC)=O)C1)CC1CCCC1 20077,Cn1cc(C(=O)NCCC2(NC(=O)C(O)C3CCC3)CC2)c(-c2cnccn2)n1 20078,C(=O)(CC(C(F)F)NC(=O)CC1CC(F)(F)C1)NCC1N(C)CCOC1 20079,C1(NC(c2ccn(CCN(C)C)n2)=O)CCC(NC(=O)CC2CCC3CC23)CC1 20080,C1(NC(C2(CCNC(c3c(C)coc3)=O)CC2)=O)CCCCC1N=[N+]=[N-] 20081,C(=O)(C(CO)C(C)(C)C)NCC1CC(CNC(Cc2nn(C)c(Cl)c2)=O)C1 20082,c1(C(N2CCC(OC)(CO)C2)C(=O)NCC)ccc(OC(F)F)cc1Cl 20083,C1(n2c(-c3ccc(CC4CC4)o3)nc(COC)n2)CCOC(C)(C)C1 20084,CC1CCCC(C(=O)NCCCOCCC(=O)NCc2ccn(C3CC3)n2)C1 20085,C(=O)(C1=CCCCCC1)NC(C)CCCCNC(=O)CNC(C1CCCCC1)=O 20086,c1(CSCC(N2CC(CC(C)NC(=O)C(C3CCCCC3)O)C2)=O)ccccc1 20087,c1(C(=O)NC2C(CNC(c3cnn(C)c3Br)=O)C2)cc(F)cc(Cl)c1N 20088,C=C(C)CC(C(=O)NCC1CC(C)=NO1)NC(=O)C=C1CCOCC1 20089,N1(C(C(CCC)CNC(C2(CC(=O)OC)CC2)=O)=O)CC2CCCCC2C1 20090,CCCCCS(=O)(=O)CC(=O)NCC1CCN1C(C1CC12CC(OCC)C2)=O 20091,C1(C(=O)NCC2CC(OC)C2)(NC(c2cnncc2C)=O)CCN(C)C1 20092,Cc1ccc(-c2nc(Cn3nccn3)n(C3CC3)n2)cc1Br 20093,N1(C(CC)=O)CC(N(C)OC)C1.c12n[nH]cc1C(=O)NC2 20094,C(=O)(CCC(F)(F)C(F)F)NC(C1CCOC1)CNC(c1c(C)cnnc1O)=O 20095,N1(C(C(COC)(C)OC)=O)CCC2(CC1)CN(C(C1(C(C)C)CCC1)=O)C2 20096,c1(C(N2CCSCC2)C)cn(CC2C=CCN2C(c2cc(C(=O)O)on2)=O)nn1 20097,N1(C(CC(C(C)C)O)=O)CCC(C2(O)CCN(C(=O)CN3CCCC3=O)C2)CC1 20098,c1(OC)c(C(=O)NC(CNC(=O)Cc2ccc(C)nc2)CO)ccnc1Cl 20099,c1(C(=O)NCC2CC(CNC(CSS(C)(=O)=O)=O)OC2)cc2ccnc(Cl)c2s1 20100,c1(C(N2CCC(N(C(C(CC)NC(N)=O)=O)CC)C2)=O)cnc(C)c(C(C)=O)c1 20101,c1(CC(=O)N(c2cccc(OC)c2)C(C)C)cccc2ccncc12 20102,C(c1c(C)noc1C)=CC(N1C(C2CCCN(C(CS(CC)=O)=O)C2)CCC1)=O 20103,C1(CNC(C2COC3(CCC3)C2)=O)CN(C(=O)C2=CCCSC2)CC12CCC2 20104,c1(C(N(C2CCCCN(C(=O)C(C)(F)C(C)(C)F)C2)C)=O)ccn2nncc2c1 20105,Cc1nnc2ccc(C(=O)NCCNC(C34CCCC3CC4)=O)cc2c1C 20106,Cc1cc(C(=O)NCC2CN(C(c3cnnc(O)c3)=O)CCCO2)cc(C)c1N 20107,CCCC(C(=O)N1CCCN(C(c2oc(SC)cc2C)=O)C(C)C1)S(N)(=O)=O 20108,C1(C(=O)NC(C)CNC(c2c[nH]nc2-c2ccco2)=O)CCNC(=O)C1 20109,C#Cc1cnc(N2CCN(C)CC2CNC(=O)Cc2ccn(C(C)C)n2)nc1 20110,CCC(C)(C)CC(=O)N(C(CC(F)F)C(=O)N1CC(N(C)C)C(F)C1)C 20111,C(CC(=O)NC1CCC1NC(c1cnns1)=O)SCC(C)C 20112,CCC(COC)C(=O)NCC(C)(C)C(=O)N(CC(C)C(=O)OCC)C 20113,N1(C(C=CC)=O)CC(C)(C)CC1C(=O)NCC1COCCO1 20114,C1(NCc2c(C)nsc2C)CC(NC(c2ccc(-c3cc[nH]n3)s2)=O)C12CCC2 20115,C(CCCOC)(C(=O)N(C)Cc1cnccc1C)NC(C(CCC)O)=O 20116,C(=O)(C1CCCc2nc[nH]c21)N(CC(C)NC(C1(C)CC2(CCC2)C1)=O)C 20117,CC1CCC(C(=O)NC2CC3(CCC3)C2O)N(C(=O)Cn2cc(CO)nn2)C1 20118,N1(CC(=O)N(C2CCCC(NC(c3ccnc(S)c3)=O)C2)C)CCNC(=O)C1 20119,c1(C(=O)NC2C(C(=O)NCCN(CC)CC)CC2)cccc(C)c1O 20120,C1(CCNC(c2cnn(CC3CCCC3)c2)=O)CCN(C(=O)CSC2CC2)C1 20121,c1(C(=O)NC(CC)CNC(=O)CCCOC2CCOCC2)c(C(F)F)cnn1C 20122,C1(F)(CNC(C(CC)=CC)=O)CCC(NC(=O)CC2(CC(=O)OC)CC2)C1 20123,Cc1ccc(OCC(=O)NC2CCCC2NC(c2cc[n+]([O-])cc2)=O)cc1 20124,c1(CN(C(=O)NCC(C2(C(=O)OC)CCC2)(C)O)CC)c(C)cccc1C 20125,c1(C(=O)NCC2CCC(CNC(=O)CCC3CC3)CC2)c[nH]c2ccncc12 20126,C1(COC)(NC(c2ccc(I)cc2)=O)CCN(C)C1 20127,c1(C(=O)NC(CCOC)CNC(=O)C(C)(C)C)ccc(OC)c(OC)c1OC 20128,CC(=O)CCN=C(NCc1ccc(Cl)cc1F)N1CCC(F)(c2ccccc2)C1 20129,C1(C(=O)NCC23OCC(NC(c4ccnc(C)n4)=O)(C2)C3)COCC(C)(C)O1 20130,c1(CC)ccc(-c2nc(C(=O)NC3CCC3CNC(=O)CSCC)cs2)cc1 20131,N1(C(C(c2cc(Cl)sc2Cl)C)=O)CCN(C(=O)C(C)(C)O)CC1C 20132,Cc1ccc(C(N2CCC(CO)(NC(=O)C(C)Cn3cccn3)CC2)=O)cc1F 20133,CC(CNC(c1[nH]nnc1C1CC1)=O)C(F)C(=O)N1CCC(F)(F)CC1 20134,C1(NC(c2n(C)cc(Cl)c2)=O)CS(=O)(=O)CC1NC(C1CCS(=O)(=O)CC1)=O 20135,c1(CC(=O)NCC(C2CCOC2)NC(C2(CC=C)CC2)=O)csc(COC)n1 20136,C#CC1(CNC(C23CC2CN(C(=O)C(C)OCC(F)(F)F)C3)=O)CCCC1 20137,N1(C(c2n(C(C)C)ccc2)=O)CCCC(NC(=O)C(C)(C)c2cncnc2)CC1 20138,N#Cc1cnc(NC(C2CCCN2C(c2cc(F)cc(I)c2)=O)=O)c(Cl)c1 20139,c1(CC#N)ccccc1C(=O)NCC1CCN(C(=O)CC2CC3C=CC2C3)CC1 20140,c1(CC(C)C(=O)NCC(Cc2ccc(Cl)cc2)CO)ccc(O)cc1 20141,CC1(C(N2CC(c3cccc(F)c3)C(N)C2)=O)CCCC1(F)F 20142,c1(OC)cc(C(=O)N(C)CCOc2sccc2NC(=O)OC(C)(C)C)[nH]n1 20143,N1(C(C(C)NC(=O)C(C)(C)C)=O)CC2CCC(CNC(=O)CCC3(C)N=N3)(C2)C1 20144,N1(C(c2c(CCC)cccc2)=O)CCC(NC(=O)CCC(C)N(C)C)C(CO)C1 20145,C(=O)(N=c1ccc(C2CCOC2)n[nH]1)c1c(Br)c(C)cc(OC)c1 20146,C1(C(=O)Nc2cnn(C3CC3)c2)CCC(C(=O)NCC2CC2Cl)CC1 20147,C1(F)(CNC(c2c(COC)onc2)=O)CCCN(C(c2csc(CO)n2)=O)C1 20148,C(=O)(C1=CCN(C(c2coc(CO)c2)=O)CC1)N1C(C(C)O)COCC1 20149,N1(C(CC)=O)CCC2CN(C(C3CC(=O)C34CCC4)=O)C2C1.C1CCC1(OC)OC 20150,C(=O)(C(C)(C)C(C)C)N(CC=C1CCN(C(C=Cc2n(CC)ccn2)=O)CC1)CC 20151,C(C(CCC)CCC)NC(CC(=C)C)CO.OC 20152,N1(C(CC(C)(F)F)=O)CCCC12CCN(C(c1cc(O)cc([N+](=O)[O-])c1)=O)C2 20153,C(=O)(C(C)(C)C1=CCN(C(=O)CN2CCOCC2)C1)NC1C(O)CCC(C)C1 20154,N1(C(c2cnc(Cl)n2C)C(=O)Nc2c(C)cc(F)cc2)CCCC2(CCC2)C1C 20155,c1(C(=O)NC(CC(C)NC(Cc2c(CC)con2)=O)C)cc2cc(Cl)ncc2[nH]1 20156,c1(C(=O)NC(CCNC(C(COC)OC)=O)(C)C)cnc2cnccc2c1 20157,C(C(COC)C(=O)NCCCCCN(C(=O)Cn1nccn1)C(C)C)OC 20158,CC1CC(CNC(=O)CCCC2CC2)CN1C(=O)CC12CCCC1C2 20159,c1(C(C(=O)NC(C)(C)C)N(CCC(=O)OC)C(C)C)nc(C(F)(F)F)n[nH]1 20160,Cc1cc(F)c(C(N2CCN(C(c3cn4ccccc4n3)=O)C3CC23)=O)c(F)c1 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20281,CCC(O)(C(=O)NCC1(COC)CCN(C(=O)CC(=O)NC)C1)c1ccccc1 20282,C1(NC(C(CC)C)=O)CN(C(=O)Cc2ccc(CO)cc2)C2(CCCCC2)C1 20283,C(=O)(C#CC1CCOCC1)NC1(C(N2CCC(C)CC2C)=O)CSC1 20284,C(CC1=CCN(C(C2(C3CCOCC3)CC2)=O)CC1)NC(C(C)(C)C(N)=O)=O 20285,c1(C(=O)NCCC2CN(C(C=CSC)=O)C2)ccccc1[N+](=O)[O-] 20286,c1(C(C)C)occc1C(N1CCCC1C1(NC(C2C3COCC23)=O)CC1)=O 20287,n1(CC)ncc(C(=O)NC(C)CNC(c2csc(-c3ncccc3F)n2)=O)c1C 20288,C1(CC)CN(C)c2ccccc2CN1C(=O)Nc1nc(CN(C)C)cs1 20289,C(=O)(C1CSc2ccccc21)NCC1(CNC(C(F)=CCC)=O)CC12CCC2 20290,CN1CC=C(C(=O)OCCCOCc2ccccc2F)C1 20291,C1(C(N2CCCC2)=O)CC2(C1)CC(CN=c1ccn(-c3nccs3)[nH]1)C2.n12nnnc1C1CC21 20292,C(=O)(CC(F)(F)F)NCC(C)(CC)NC(c1ccn(CCC)n1)=O 20293,C1(C(=O)NCc2ccc(-c3cccc(C)c3)cc2)COCC(=O)N1C(C)C 20294,n1(CC)ncc(C(=O)N(CCCN(C)CC2CCOCC2)C)n1 20295,Cc1cccc(CNC(=O)CC(C(C)C)NC(c2cncn2C(C)C)=O)c1C 20296,C12(COC)CC(NC(=O)C(Cc3ccco3)NC(=O)Cn3cc(CO)nn3)(CO1)C2 20297,c1(C(C(=O)N(C)CC2(NC(c3cn(CC=C)nc3)=O)CC2)(F)F)cccc(C)n1 20298,S(=O)(=O)(c1ccc(Cl)cc1F)N1CC(F)CC(C(N2CCCOCC2)=O)C1 20299,C1(COC)(NC(=O)C(C)OCCc2ccccc2)CCN(C(=O)C(C)OC)CC1 20300,CN1CCN(C(c2cnc(C3CC3)nc2)=O)C(CNC(C2CCC3CC3C2)=O)C1 20301,Cc1nc2c(NCc3ncccc3C(=O)O)cccn2n1.c12cc(ccc1O)OC2 20302,Cc1ccccc1OCC(=O)NC1(CF)CC1 20303,N12CC(C3(CC3)C1)C2=O.N1(C(COCCOCC)=O)CC(C)C1.N(C)C 20304,C1(C(N(C)CCOCC2CC2)=O)CC(C)(C)CCN1C(c1cnccc1C#N)=O 20305,C(C(C)(C)CC(=O)NC1(CC(=O)N(C2CC2C)C)CCCCC1)OC 20306,C(C(=O)N(CCCCO)C)(C(C)OC)NC(CCOCC#C)=O 20307,c1(C(N2CC(NS(C)(=O)=O)C2)=O)csc(Cl)n1 20308,C1(NC(c2cc(C(C)C)ncc2)=O)CN(C(C2CCCCO2)=O)CC1(F)F 20309,O=C(C1=CN=C2N=CNN2C1)N1CCCC1C1CCN(C(=O)C(O)C2CC2)C1 20310,CCC(CC(=O)NCC(CC(=O)Nc1ccc(CO)nc1)C1CCC1)OC 20311,C1(C(N(C(C(C)C)CO)C)=O)C2CC3C(C2NC(c2c[nH]c(=N)o2)=O)C13 20312,c1(C(=O)NCCN(C(=O)C(CO)OC)CCOC)ccc(C#N)cc1O 20313,c1(CC(=O)N(C(C)C)CCNC(C2(CCF)CC2)=O)ccco1 20314,c1(CC)nc(C(C)C)ccc1CNCCC12CCC(C)(C1)OC2 20315,c1(C(=O)OC)cc(=NC2CCCC(NC(=O)CCCCCC(C)(C)C)C2)[nH]c(Cl)n1 20316,Cc1cc2n(n1)CCN(C(=O)CC1CN(C(=O)CSC(F)F)CCC1C)C2 20317,c1(C(=O)NC(c2cccc(Cl)c2)CNC(C2(CC)CC2)=O)cnc2scnc2c1 20318,c1(C(=O)NCCNC(C2CC(=C)C2)=O)cc(Br)c(C)o1 20319,c1(C(c2n(CCC)nnn2)NCc2nc(C)n(C)n2)ccc2c(c1)OCC(=O)N2 20320,Cc1ccc(C(=O)NC2(C(=O)NC3CCOCC3C)CCSC2)nn1 20321,c1(C(=O)NC2CCC(CNC(c3cnc(C(C)=O)s3)=O)C2)cc(C)c(Cl)cc1C 20322,C(C(O)CS(C)(=O)=O)N(C=O)Cc1c(C)nn(Cc2ccccc2)c1 20323,CCCCC(C(=O)NCCCOC)NC(c1cn(CC)nc1C)=O 20324,Cc1cccc(C(N2CCC(F)CC2C(=O)NCCN2CCCC2)=O)c1O 20325,N(C1CCC(NC(=O)Cc2ccccc2O)c2ccccc21)C(=O)C=CCF 20326,c1(C(=O)NC2C=CCN(C(Cc3c(C)scc3)=O)C2)cccc(Cl)c1C 20327,Cc1nc[nH]c1CC(=O)N(C1CCC(NC(=O)Cc2cnc[nH]2)C1)C 20328,CON=CC(=O)NCCCC(=O)NCCNC(=O)C1CC1 20329,C(CNC(=O)Cn1nccc1C(F)F)(CCCC)NC(CCCNC(C)=O)=O 20330,C12(CNC(c3c(C)noc3)=O)CCCC1CN(C(c1cnc(N(C)C)o1)=O)C2 20331,C#CC1(C(=O)NC(CC)CCCCC)CCN(C(C2C3CCC(C3)C2C)=O)CC1 20332,C1(NC(c2c(C)coc2C2CC2)=O)CC(F)CN(C(C2CCCOC2)=O)C1 20333,Cc1nc2nccc(NC3CC(F)(F)CC3C(=O)OC(C)(C)C)n2n1 20334,Cc1[nH]c(=N)sc1CNC(=O)C(=O)N(CC1CC1)CC1CCCNC1 20335,C1(NC(=O)C=Cc2ccc(Cl)cc2F)COC2(CCN(C(=O)CC3(O)CC3)C2)C1 20336,C1(CNC(C2CCC(C)(CC)O2)=O)CN(C(=O)CSc2nncn2C)CCN1C 20337,c1(C(=O)NC2C(CO)CCN(C(c3c(CC)ccs3)=O)C2)cc(S(C)(=O)=O)co1 20338,Cc1cccc2c1CCCC2NC(C1(C)CCC(=O)N1)=O 20339,N1(C(CC(n2ccc(C)n2)C)=O)CCCCC12CC(NC(=O)CC(C)CF)C2 20340,CCC(CC)CC(=O)NC(CNC(=O)CC1CCCN1C)C(C)C 20341,N1(C(=O)OC(C)(C)C)CC2(C1)CC1(CC(NC(=O)Nc3ccc(I)cc3)C1)C2 20342,N1(C(CC(C=C)CC)=O)CC2(C(=O)NOCCC(F)(F)F)CC1CCO2 20343,CC1(CNC(=O)CCOCC(F)(F)F)CCN(C(C2CCCC(F)C2)=O)C1 20344,Cc1cc(C(=O)NCC2CN(C(=O)CN3CCCS3(=O)=O)C2)ccc1Cl 20345,N1(C(C(c2n(C)ccc2)=O)=O)CC2(CCCC(CNC(=O)Cc3cnns3)O2)C1 20346,C=CCCC(C(=O)NCC1(C)CCCO1)NC(c1ccccc1Cl)=O 20347,c1(CC)ccc(C(=O)NC2(CNC(=O)CC3CC34CC4)CCCC2)cn1 20348,C1(N(C2CC(CC(=O)O)(CO)C2)C(C2(c3cn(C)nc3)CC2)=O)CCC(F)(F)C1 20349,CS(C)(=O)=NC(=O)C(=O)NC12CC(CNC(=O)CCc3cn[nH]c3)(C1)C2 20350,C1(CCNC(c2cnn(CC3CC3)c2)=O)CC(F)(F)CN1C(=O)Cc1ccno1 20351,N1(C(c2c(N)ccc(C)c2)=O)CC(NC(=O)CC2OCCCO2)C2CCCCC12 20352,CCCCC(C(=O)NCC(C1CCCCC1)NC(=O)C(F)F)NC(N)=O 20353,c1(C(=O)NCC(C)NC(C2CC(C(C)C)C2)=O)ccc2cc(O)ccc2c1 20354,Nc1cc(C(=O)NCC2CC2CNC(C2(n3nccn3)CC2)=O)cc(O)c1Cl 20355,C(C(C(C)C(C)C)NC(=O)Cc1ccc(C)cc1)NC(c1ccc(CCC)[nH]1)=O 20356,CC1(Cn2cc(CCN3CCSCC3)nn2)CCCCC1(F)F 20357,C#Cc1ccc(C(N2CCC(C(=O)NCC(O)COC)(CC)C2)=O)o1 20358,N1(C(c2cc(F)cc(Br)c2)C(=O)NC)CCC2CCCCC12 20359,c1(C(N2CCCCC(NC(c3ccc(C)s3)=O)C2)=O)cc(Cl)c(N)cc1F 20360,c1(-c2n(CC=C)c(N(CC(C)C)CC)nn2)ccc(S(C)(=O)=O)cc1 20361,C(=O)(C#Cc1ccccc1)NC1C(C(=O)NC2CCN(C(=O)OC)CC2)CCC1 20362,c1(C(C)C)ccccc1C(=O)NC1CC1CNC(=O)C=C1CC1 20363,C1(NC(C(CSC)(C)NC(=O)Cn2cnnc2)=O)CCN(OC)CC1 20364,N1(C(CC(C)SC)=O)CCCC(C(=O)NCC2(n3ccnn3)CC2)C1 20365,N1(C(CN(C2CC2)CC)=O)CC2CC(C(=O)NCc3cnc(C)cc3C)(C2)C1 20366,CN=c1nc(N2CCC(C)(CC#N)C2)[nH]c(=NCC2(c3ccccc3C)CC2)[nH]1 20367,c1(C(N2CC(C)C(CCNC(=O)CCS(C)=O)C2)=O)cc(F)c(F)c(C#N)c1 20368,c1(C(N2C(C(=O)Nc3ccc(CCO)cc3)CC(C)C2)=O)c(F)cc(Cl)cc1Br 20369,C1(CNC(CSCC(=O)OC)=O)CC2CCC1N(C(=O)C(C)C1CCOC1)C2 20370,C(=O)(CC1=CCN(C)CC1)NC1CC2CN(C(c3c(NC)cccc3)=O)C(C1)C2 20371,n1(CC)cnc2c(N3CCC(C(C)O)C3)nc(N(CC(C)(C)CO)C)nc12 20372,C1(NC(c2cc(COC)[nH]n2)=O)CCCCC1CNC(=O)Cc1ccns1 20373,CN1CC(CC(=O)NCCOCCN(C(=O)CC=C(Cl)Cl)C)C(O)C1 20374,c1(C(=O)NC(C(C)C)CNC(C2(C)C=CCC2)=O)cc(F)c2c(c1)CCC2 20375,N1(C(Cc2cc(C)nn2C)=O)CCCC(C)(C(=O)Nc2cccnc2C(C)C)C1 20376,C1(CCCC)CCCN1C(=O)C(C1CCC1)NC(=O)C=CCC1CCCC1 20377,c1(CC)cc(N2CCCC(NC(C3CCC(=O)N(C)C3)=O)C2C)nc(CC)n1 20378,CCC(CC(=O)N1CC(C2CC2C(=O)N(CC(C)C)C)C1)C(C)(C)C 20379,C1(NC(C(C)OCC)=O)CCCCN(C(C2(C)CCN(C)CC2)=O)CC1 20380,C(=O)(C1CCCc2nc[nH]c21)N1CCC(NC(=O)C=Cc2cscn2)C12CC2 20381,CCCCCCCCCCCC(=O)N(CC(CC)NC(C1(OC)CCSC1)=O)C 20382,C1(NC(c2cc(CC)c(OC)cc2)=O)C2CC(CN(C(C3(O)CC3)=O)C2)C1CO 20383,Cc1cccc2c(CC(=O)NC3COCC3NC(C3CC4(CCC4)C3)=O)c[nH]c12 20384,C1(CC#N)CCCN1C(=O)Cn1nnnc1Br.c1ccccc1 20385,N1(C(C2(COC)CCC2)=O)CC2CC2(CNCc2cnc(C3CC3)s2)C1 20386,C(CC1=CCN(C(C2CC(=O)OC2(C)C)=O)CC1)NC(CC(C)CN(C)C)=O 20387,C1(CC(=O)NC(c2nc(C)cs2)CC)CN(Cc2ccc(C(=O)O)s2)CCO1 20388,Cc1cc(CC(=O)NC23CC2CN(C(=O)CSc2cn[nH]c2)C3)nn1C 20389,N1(C(C(CC)C#N)=O)CC2CCOC2(C(=O)OC)C1 20390,C1(CC(=O)NC)CCN(C(=NCc2cc(Cl)ccc2O)NC2CC2C)CC1 20391,CC1CCCN(C(c2c[nH]c(=O)cn2)=O)C1CNC(=O)C(O)Cc1cnc[nH]1 20392,Cc1ccc(C(F)(F)C(=O)NC2CCC(NC(C3CC(=O)N(O)C3)=O)CC2)cc1 20393,c12cc(Br)c(nc1C)C(=O)C2N1CCN(c2cc(C)ccc2C)CC1.CN 20394,C=CCCCC(C(=O)NC1CNC(=O)C1(C)C)NC(c1nc(C)oc1C)=O 20395,O=C1NCCCCC1NC(c1ccc(I)cc1)c1nnnn1CCCF 20396,N1(C(C(CN(C)C)O)=O)CCC(N=[N+]=[N-])(C(=O)NCc2ccoc2)C1 20397,Cc1cc(NCC2(F)CCCC2)ncc1S(=O)(=O)NC1CCC2C(CC1)C2(F)F 20398,O=C(CC1=CSC2=NCCN12)N1CCC(O)(CO)CC1 20399,c1(OC)ccc(C(N2CC(O)(C(C)NC(=O)C(O)Cc3[nH]cnc3C)C2)=O)o1 20400,CCC(C(=O)N1CC2CC1(C(=O)NCCC1(COC)CCC1)C2)C(F)(F)F 20401,c1(CC)occ(C)c1C(=O)NCC1CCCC(NC(C2(N=[N+]=[N-])CC2)=O)C1 20402,c1(C(N2C(C(C)(C)NC(c3c(CC)cns3)=O)CCC2)=O)cn2cnnc2cn1 20403,CN1CCN(C(=O)Cc2n[nH]c(=N)s2)CC1CNC(C1CCCCC1CO)=O 20404,C(CC(=O)N1CCC(OC2CCC2)C1)(C(F)(F)F)NC(C(F)=CCC)=O 20405,C1(NC(c2c(C)n[nH]c2)=O)C2CCN(C(=O)C=CC(=O)NC3CC3)CC12 20406,Cc1ccnc(CS(=O)Cc2ccccn2)c1Br 20407,Cc1cccc(CC(=O)NCCC2CCCCN2C(=O)Cc2cccnc2)c1 20408,c1(C(=O)NC(c2ccc(C)cc2)c2ccccn2)ccc(F)c(C)c1Cl 20409,N1(C(C2(CC=C)CC2)=O)CC2(CO)CC1(C(N1CCOC(C3CC3)C1)=O)C2 20410,CC1CN(C(C2CC(O)C2)=O)CC(C)C1NC(c1nnn2c1CSCC2)=O 20411,N1(C(C(CC)F)=O)CC2CCC(NC(=O)C3=CCOCC3)CC2C1 20412,c1(C(=O)OC)no[nH]c1=NC(=O)c1nc(C(=O)Nc2csc(C)n2)cs1 20413,C1(N(C(CC)=O)C)CCCC(NC(c2cn(CCOC)nc2C)=O)C1 20414,c1(C(=O)OC)ncc(Br)c(OCc2ccccc2)n1.C12CC3CC(C3C1)N2 20415,c1(CN2C(C(=O)NCCc3ccco3)C(O)CC2)c(F)ccc2occc12 20416,O=C(C#CC1CCCC1)N1CCN(C(c2cc[nH]c2C2CC2)=O)C(C2CC2)C1 20417,S(=O)(=O)(C1CCCCC1)N1CCN(C(C2(C)CCN(C(=O)OC(C)(C)C)C2)=O)CC1 20418,C1(C(=O)NC2CCCC(C(N(CCCC(C)C)CCO)=O)C2)CC2(C1)CC(O)C2 20419,C1(C(N(CCCC(=O)NC)C)=O)C(C2CC2)CCN1C(C1CCCC1)=O 20420,C1(CNC(C(C)(C)F)=O)CC2(CCN(C(c3cnc(C#N)s3)=O)CC2)C1 20421,C1(C(=O)NCCC2CCN(C)CC2)CC(N=[N+]=[N-])CN1C(C1C2CN(C)CC12)=O 20422,C1(NC(CC(=C)C)=O)CN(C(C2(c3ccc(F)cc3F)CC2)=O)C2(CCOC2)C1 20423,c1(CC2CCN(C(c3cc(Cl)ccn3)C(=O)NCC(C)C)C2)ccc(F)c(F)c1 20424,N1(C(c2c(CC)nc[nH]2)=O)CCC2(C1)CN(C(=O)C(C)C#N)C2 20425,N#Cc1ccc(C(=O)NC2CC2CNC(C2CCS(=O)(=O)C2)=O)o1 20426,CC(CN(C)C)CCC(=O)NCC(O)CNC(C12CCC(CC1O)C2)=O 20427,c1(C(=O)NCCN(C(c2nccc(OC)c2F)=O)CC)cnn2c1CCC2 20428,C#CCCCC(C)C(=O)NCc1ccc(CNC(=O)C(C)(C)OC(F)(F)F)cc1 20429,c1(C(N2CC(OCCC(=O)NC(CCC)CC)C2)=O)cc2occc2[nH]1 20430,N1(C(CN2CC(C)C2)=O)CCOC2(CCN(C(=O)C3=CCCCCC3)C2)C1 20431,c1(OCC)cnc(C(=O)NC2CCC2NC(c2ccon2)=O)cn1 20432,C#Cc1ccc(C(=O)NC2CCCCN(C(c3scnc3CC)=O)C2)cn1 20433,c1(OC)cc2cc[nH]c(=O)c2s1.c12ccccc1-c1cn(nn1)CC(=O)N1CC2C1 20434,CC1C(NC(=O)C(C)NC(N)=O)CCCN1C(C1CC12CCCC2)=O 20435,C1(NC(CCN(C(C(CC)CCOC)=O)C2CC2)=O)CCN(C)CC1(C)C 20436,c1(C2(C(=O)NCC(C)(F)CNC(=O)Cn3cc(Cl)cn3)CC2)cccnc1Cl 20437,N(C1CCCc2cccc(F)c21)S(c1ccc(CC(C)C)o1)(=O)=O 20438,N1(CC(C)C)CC(NS(=O)(=O)CC2(C)CC2(F)F)CC1=O 20439,N1(C(C(=O)NCCOC)=O)CCCC(C(=O)NCC23CC(C2)C(C)O3)C1 20440,c1(COC(CN(C(=O)Cc2ccc(Br)s2)CC)=O)ccc(C#N)cc1 20441,C=CCC(C)(C)CC(=O)NCc1ccccc1CNC(C1NC(=O)CC1C)=O 20442,N1(C(=O)OC(C)(C)C)CCC(NC(C2C(=C)C2NC(=O)CC2CC2)=O)C(O)C1 20443,O=C(N=c1nc(Cl)nc2[nH][nH]cc1-2)C1CN(C(c2ccncc2O)=O)CCO1 20444,C1(CC)CCCC1(C)C(=O)NC(C1CCN(Cc2ccsc2)CC1)C 20445,C12(NC(c3cccc4nonc34)=O)CCCN(C(C3CC(F)(F)C3)=O)CC1C2 20446,Cc1cc(C(N2CCC(CCNC(c3csc(Cl)n3)=O)CC2C)=O)nc(C)n1 20447,N1(C(N2CC(OC)CC2(C)CO)=O)CC2(CC=CCO2)C1 20448,Cc1cc(F)c(NC(CNC(CC2CC2(F)F)C(=O)OC(C)(C)C)=O)nc1Br 20449,c1(OC)cc(Br)c(CN2CCCC2CCC(=O)Nc2ccnc(F)c2F)cc1O 20450,c1(CC)[nH]ccc1C(=O)NC(C)(CNC(=O)C1CC1)C1CC1.C12CCCN1C2=O 20451,Cc1ccc(N2CCC(=O)NC2=O)cc1NC(c1cc(CC(C)(C)O)ccn1)=O 20452,C1(NC(C(C)C(F)F)=O)(CNC(c2cnn(C3CC3)c2)=O)Cc2ccccc2C1 20453,c1(-c2cn(CCC)nc2)nc(C(=O)N(Cc2ccccc2Cl)CC2CC2)c(C)s1 20454,CC(C)C(C(=O)N(C)CCOCCN(C(=O)CC1CCCC(=O)C1)C)NC=O 20455,N1(C(C2(OC)CCN(C(c3scnc3C)=O)C2)=O)CC(C)(C2CCC2)C1 20456,C1(CNC(c2ccc(SC)s2)=O)CC(NC(=O)Cc2cncnc2)C12CCC2 20457,C1(O)(CN(C)C(c2ccc(C(C)(F)F)cc2)=O)CCN(C(C2CC2F)=O)C1 20458,N1(C(c2c(C)ncn2O)=O)C2CCC1CN(C(c1cc(CO)ccc1Cl)=O)C2 20459,c1(COC)cccc(OC(c2nn[nH]n2)C)c1.c12nc(cs1)C(=O)OC2C 20460,N1(C(C=C(CCC)C)=O)CC(NC(c2ccc(O)cc2)=O)CC1(C)C 20461,C1(N(C)C(c2coc(Cl)c2)=O)CN(C(c2csc(CC(F)F)n2)=O)CC1F 20462,c1(OC)ccc(-n2nnc(C(=O)NC(C)C(CO)NC(=O)CC(C)F)c2C)cc1 20463,c1(C(=O)NC2(C)CCCN(c3cnc(C#N)cn3)C2)cc2n(n1)CC1(CC1)C2 20464,c1(C(c2nnnn2C)Nc2ccc(OCCC)cc2C)ccc2c(c1)CCC2 20465,C1(C(N2CCC(C(=O)NCCOCCC=C)(CF)C2)=O)CCCC2(CC2)C1 20466,CCCC(O)C(=O)N1CC(N(C(=O)C(CCO)N(C)C)C)C1 20467,C1(N(C(=O)CCCc2sccc2C)CC)CCCN(C(C2CCCCC2)=O)C1 20468,C#Cc1cccc(CNC(C2CCCCN(C(=O)CC3CCCC(C)O3)C2)=O)c1 20469,C1(CNC(C(CC)C(C)C)=O)CC2(CCCN(C(=O)COCCCF)CC2)C1 20470,N1(C(c2n(CC)ccn2)=O)C2CCC1CC(C(=O)Nc1cnn(CC(N)=O)c1)C2 20471,c1(C(=O)NC(C(=O)NCCOC)C2CCCO2)cnc(O)c(F)c1 20472,O=C1CC(C(=O)N2CCCOCC23CCC3)c2ccccc21 20473,C1(CC)CCN(C(=O)CSC(F)F)C(C(=O)NOCC(C)C(=O)OC)C1 20474,c1(C(=O)NC2C(NC(c3onc(C)c3C)=O)CCC2)ccc2c(c1)COC(=O)N2 20475,c1(C(=O)NCC(COC)N)cc(F)ccc1NC(=O)C(C)C 20476,c1(OCC(=O)N(CC(C)CNC(=O)CNS(C)(=O)=O)C)ccc(C#N)cc1Cl 20477,C1(CC(=O)NCC2CC(C(N3C(CCC#C)CCC3)=O)C2)CC(O)C1(C)C 20478,NS(=O)(=O)CCC(=O)NCCC1CCN(C(=O)CN2CCN(C3CC3)C2=O)CC1 20479,CCCC(CC(C)C)C(=O)NC1CCN(CCCNC(=O)C#CC(C)C)C1 20480,c1(NC(=O)CN2CCCC2C(c2cccc(Cl)c2)O)ccccc1OC(F)(F)F 20481,N1(CCOCCC(=O)NCCCC)C2CCC1CCC2.C(C(F)(F)F)CC(O)CC 20482,N1(C(C2(CNC(C(C)N(C)C)=O)CC=CC2)=O)CCCNC(=O)C1 20483,c1(OC)ccc(C(=O)NCC2(NC(=O)CC3CCC(=O)C3)CCCC2)cn1 20484,C=C=C(C)CC(=O)NCC(O)C(=O)N(CCCCC=C)C 20485,c1(C(=O)NCC2CN(C(C3C4CCCC34)=O)CC2(F)F)scc2c1CCCC2 20486,c1(OC)cc(C)c(CC(N2CC(N3CCN(C(=O)CN)CC3)C2)=O)cc1F 20487,N1(C(CC(C)F)=O)CCCCC12CN(C(=O)C(F)(F)c1csc(=N)[nH]1)C2 20488,C1(C(=O)NCC2(OC)CN(C(=O)CC3(O)CCCCC3)C2)CCCC(C)(C)O1 20489,C(=O)(C1=CCc2ccccc21)NC(C)CCNC(c1sccc1S(N)(=O)=O)=O 20490,C1(NC(CSc2ccc(OC)cc2)=O)CCN(C(=O)CCCCCBr)CC1F 20491,c1(C(=O)NC2CC3CN(C(c4c(Cl)nc(OC)s4)=O)CC32)cncc2nc[nH]c12 20492,Nc1cc(C(=O)NCC2COCC2NC(C2(O)CCC2)=O)c(F)c(F)c1F 20493,C1(NC(C2(C)CCN(C)C2)=O)CC2CC(NC(c3occc3C3CC3)=O)C2C1 20494,c1(C(=O)NCCC2(O)CCCN(C(C(C(C)O)(C)C)=O)C2)cccn2nccc12 20495,C(c1ccc2c(c1)OCO2)=CC(=O)NC1(CNC(C(CCCC)C)=O)CCOC1 20496,C1(OC)CC(CC(N2CC(N(C(=O)CCN3CCC(C)CC3)C)C2)=O)C1(C)C 20497,c1(C(=O)OC)ccc(OC)c(F)c1NC(C1CSC(Cc2ccccc2)C(=O)N1)=O 20498,c1(C(N2CC(F)(CNC(C3CCC(CC)C3)=O)C2)=O)ccc(OC)c(Cl)c1OC 20499,c1(OC)c(C(=O)NCCC2(O)CN(C(C3CCCC(F)C3)=O)C2)c(C)nn1C 20500,C12(C(=O)NCc3ccc(C)nc3O)CCC(CN(C(=O)C(F)CC(C)(C)C)C1)C2 20501,c1(C(N2C3C(NC(C4C(CC)C4)=O)C(C3)C2)=O)ccc(S(=O)(=O)CC(N)=O)cc1 20502,c1(C(=O)NCC(C(C)C)NC(Cn2c(C)nnn2)=O)ccc(N=S(C)(C)=O)s1 20503,C(CNc1ccc(-c2ccc(Cl)cc2)cc1F)(CS(C)(=O)=O)OC 20504,C1(CCC(=O)NCCOCC#C)CCN(C(=O)Cc2cncnc2)C1(C)C 20505,C1(CNC(=O)C=Cc2cc[nH]c2)CC2CCC1N2C(C1(CO)CCOCC1)=O 20506,FC1(F)Oc2ccc(C(c3nnnn3C3COC3)NCCC3CCOC3)cc2O1 20507,c1(C(N(C2CCN(C(CCCC#C)=O)CC2C)C)=O)ccc2cccnc2c1 20508,c1(C(=O)NCC2(O)CCCN(C(c3c(C)cnnc3)=O)C2)cc2ncccc2o1 20509,Cc1c([N+](=O)[O-])c(C(N2CCC2Cn2cc(Cc3ccccc3)nn2)=O)nn1C 20510,CCCC(C(O)C(=O)N1C(C)CC1(C)C)NC(c1sncc1C)=O 20511,C(C)(CO)(C(=O)NC1CCOC(C(=O)NCC(C)CC2CCCC2)C1)OC 20512,c1(N2CCC(C(C)NC(C3CCCN3S(C)(=O)=O)=O)C2)ccc(C#N)nc1 20513,CCCC(O)C(=O)N1CCC(OC2CN(C(C3COCCN3C)=O)C2)CC1 20514,C12(C(=O)NC3(C)CC(O)C3)CC(CO)(CN1C(C1(C#N)CC3CC3C1)=O)C2 20515,C1(C(=O)NCC2CC(F)(CNC(=O)C(O)CSC)C2)(OC)CCOCC1 20516,c1(C(=O)NCCN(CCOC)C(c2c[nH]cc2Br)=O)scc(C)c1Cl 20517,CN1C(=O)CN(CC(=O)NC(CNC(=O)CCc2cc(Cl)no2)C2CC2)C1=O 20518,N1(C(C2(CC)CCC2)=O)CC2CC2(CNC(C2(CCOCC)CCOC2)=O)C1 20519,N1(C(C(C)OCCC=C)=O)CC(CNC(=O)C(C)OC2CCCC2)(SCC)C1 20520,n1(CCCC(=O)NC2CC(F)(CNC(COCCCC#C)=O)C2)c(C)csc1=O 20521,N1(C(CC(CC)(F)F)=O)CC2(CCN(C(C3CCCS3)=O)CC2)C1C(C)C 20522,C(CCSC)(C(=O)N(CC(C)N(C(=O)C=Cc1scnc1C)C)C)OC 20523,n1(CCCC(=O)NCCN(C(C2CCCC2)=O)C2CC2)cnc2ccccc12 20524,Cc1c(NCc2ccccc2)ncnc1N1CCCC(N2CCCCC2)C1 20525,N1(C(c2cnc(C)n2C)=O)CCC(n2cccn2)(C(N2CCSC2(C)C)=O)CC1 20526,CC1CC(C(N2CCC(C)(CNC(c3cnn(CCF)c3)=O)C2)=O)CCO1 20527,C1(NC(c2ccccc2C(F)(F)F)=O)CCN(C(c2nccs2)=O)CC1F 20528,N1(C(C2CN(CC)C(=O)C2)=O)CCCC2(C1)CN(C(=O)CC1CC(C)C1)CCO2 20529,c1(C(N2CC(c3cnc4ccc(F)cn34)C2)=O)ccc(=O)n2c1CCC2 20530,C1(OC)C(NC(=O)CNC(=O)CN2CCC(C)CC2)CC1(C)C 20531,C(=O)(CC1CCCc2cc(OC)ccc21)NC1CN(C(C=CC)=O)CC1(C)C 20532,c12cn(C)nc1C(c1nnnn1C(C)(C)C)C2(C)CCC.CC(CCC1CC1)N 20533,CCC(C(=O)NCC(C)(C)CN(C)C(C1CC12CC2)=O)n1ccnc1 20534,N1(C(C2(CC#C)CCC2)=O)CCC(NC(=O)CNS(N)(=O)=O)C2(CCC2)C1 20535,CC(C)CCCCC(=O)NC1CN(C(C2CC(c3cccc(F)c3)C2)=O)CC1O 20536,c1(CNC(C(C(C)C)O)=O)cnn2c1CN(C(=O)Cn1cnnn1)CC2 20537,C1(C(N2C(CN(C(C3CC(=C)C3)=O)C)COCC2)=O)OCCCC1(C)C 20538,C=C=C(C)C(=O)NC(c1cn(C2C(N(C)C)CCC2)nn1)C(C)C 20539,C(C(=O)NCCC1CCCN(C(c2n[nH]cc2Br)=O)C1)(C(F)(F)F)OC(C)=O 20540,C1(C)(CN(C(CC2OCC(C)(C)C2)=O)CC)CCC(O)CC1.C12(CCC1)C(=O)N2 20541,N1(C(C(N(C(c2ccn(CC)n2)=O)C)C2CC2)=O)CC(N(C)C)C(F)C1 20542,Cc1cc(F)ccc1N1CCCC(NC(N2CCC3CC23)=O)C1 20543,N1(C(C2CCCN(CCC)C2)=O)CCN(C(c2cnc[nH]2)=O)CC1C(F)F 20544,C1(NC(=O)CCSc2ccccc2)CCCC12CCN(C(=O)CCOC1CC1)C2 20545,CC1(C)CN(C(=O)C2=COCC2)CC1NC(C1C2CCCC12)=O 20546,N1(C(C(C)NC(=O)NC)=O)CCC2(CC1)CC(NC(=O)Cc1cocn1)C2 20547,C=CCC(F)(F)C(=O)N1CCC(F)(CNC(C2(C)CC(F)C2)=O)CC1 20548,C(=O)(C(C)(F)C(F)(F)F)NC(CC)CNC(c1cccc(N(C)C)c1)=O 20549,Cc1ccc(C(N2CCCC2C(C)(C)C(N2CC3CCC(C2)O3)=O)=O)c(O)n1 20550,c1(C(N2CCC(NC(=O)C=Cc3ccncn3)(C)C2)=O)ccc(Cl)cc1O.C 20551,CCC(CC(=O)NC(CCO)C(F)F)N(C)C(C1CC(C)(CC)C1)=O 20552,C1(C(=O)NCC2(CNC(CNC(CC(C)C)=O)=O)CCC2)COCC(C)O1 20553,c1(C(=O)NCC(CC=C)NC(=O)C=Cc2ncc(C)[nH]2)ccc(Br)cc1N 20554,C(=O)(C(O)CC(F)(F)F)NC(C(=O)NCC(COCC)(C)C)CCN(C)C 20555,c1(OCCC(=O)NCC(CO)NC(CC(C)N(C)C)=O)ccc(F)cc1 20556,C1(C(=O)NCC2C(CC(=O)N(C(CC)CC)CCO)C2)CNC(=O)O1 20557,c1(CCNC(C(CC2CC2)NC(C(COC)C)=O)=O)ccccc1F 20558,c1(C(N2CCC(N(C(C3CNC(=O)N3)=O)CC)C2)=O)cc2cccnn2c1 20559,C1(C(N(C2CCC(NC(C3(CO)CCCO3)=O)CC2)C)=O)C2CC3C(C2=O)C13 20560,C(=O)(C1=C(Cl)CCOC1)N(CCCNC(=O)CCCOc1cccnc1)CCO 20561,C1(NC(c2ccc(C)nc2O)=O)COC2(CCN(C(C3COC(=O)C3)=O)CC2)C1 20562,N1(C(C2CC(O)(CNC(C(CCN(C)C)O)=O)C2)=O)CC2CC=CCC2C1 20563,c1(NC(=O)NC(C)Cc2cccc(C#N)c2)ccc(C(N)=O)c(Cl)c1Cl 20564,CC1CN(C(c2csc(C3CC3)n2)=O)CC1CNC(C1(n2cccn2)CCC1)=O 20565,C(=O)(C#CC1CCC1)NCCCC(=O)NCC1CCC(C)C1 20566,C1(C(N2CCC(CC(=O)OC)C2)=O)CC12CCN(C(C13CCCN1CCC3)=O)CC2 20567,c1ccc(C2SCCS2)cc1.C1(C(=O)NC(C)CNC(C2CC2)=O)(OCC)CCC1 20568,c1(C(=O)OC)cc(C)c(C(=O)NC(C)CNC(=O)C(C)(C)c2ccnn2C)o1 20569,CCC(C)CCCCC(=O)NCCC1CSCCN1C(=O)C1=CCC(C)CC1 20570,N1(C(c2sc3ccn(C)c3c2)=O)CCC2(CCN(C(c3cc(F)c[nH]3)=O)C2)C1 20571,C1(CNC(C(CN(C)C)N(C)C)=O)CCC(NC(C2(C)CCCS2)=O)CC1 20572,C12(C)CCCN(C1)C2=O.C1(NC(COC)=O)CCN(C(=O)C(C)C)CC1 20573,CCCC(CCC)NC(=O)C(C1CN(C(=O)C(O)CN2CCCC2)C1)SC 20574,C12(CC)CCC(C(=O)NC3CCN(C(c4sncc4C)=O)CC3F)(CO1)C2 20575,N1(C(CCC=CC(C)C)=O)CCC(N=[N+]=[N-])(C(=O)NCC2CC23CC3)C1 20576,c1(C(N2CC3C(NC(C4(CC=C)CCCC4)=O)(C3)C2)=O)c(C)nc(O)nc1C 20577,C1(CNC(C2(C)ON=C(C)C2)=O)CC2(CO1)CN(c1cc(O)nc(O)n1)C2 20578,CC1CN(C(c2ccnnc2)=O)CC2(CCN(C(=O)Cc3cn[nH]c3)C2)O1 20579,c1(C(=O)NC(CCN(C(C(C(C)C)OCC)=O)C)C)sc(Cl)c(Cl)c1OC 20580,C1(NC(c2nc(C)oc2C)=O)CC(C)CN(C(=O)CC2(C)CCC2)C1 20581,S(=O)(=O)(c1ccc(C(=O)N(C2CN(C(C3(C)COCCO3)=O)C2)C)cn1)NC 20582,C1(CNC(=O)C(F)CC2CC2)CC2COCC2N1C(=O)CCCCCO 20583,C(=O)(CCC1=CCCCC1)NC1(CO)CCCN(C(CCN(CCC)C)=O)C1 20584,N1(C(=O)CN2CCCC2=O)CCCC2CN(c3cc4nncn4cn3)CC12 20585,C1(C(=O)NCCc2onc(C)n2)CC2CC1CC2NC(=O)C(C)CN(C)C 20586,C1(CCC(=O)NC)CCCCN1C(C(=O)NC1CCOCC1)C1CC1C 20587,C1(CC(=O)NC2(CC#C)CCN(C(COCC#C)=O)CC2)COCC2(CCC2)O1 20588,C1(C(N2CC(CNC(COC)=O)C(C)C2)=O)CCCCC1C1CC1 20589,C1(C(N(CC#C)C2CC2)=O)CSCN1C(C1CCCC1O)=O 20590,c1(CC)ccc(C(=O)NC2CCC2NC(c2cccnn2)=O)cc1CC 20591,c1(CN=C(NC2(CO)CC(C)(C)C2)NC2CCCC2)ccc(O)cc1Cl 20592,Cn1nc(C(=O)NCC(C)(C)NC(=O)CC2CCC3CC23)cc1C(F)F 20593,CCCCCCCC(=O)N1C2CCC(C2)C1CNC(c1ncccc1C(N)=O)=O 20594,C1(CCOC)(NC(=O)C(F)=CC2CC2)CCN(C(c2cnc(C)n2C)=O)C1 20595,c1(C(C)C)noc(Cn2cc(C3CC3C(=O)N(C(=O)CSn3cncn3)C)nn2)n1 20596,CCS(=O)(=O)CCCNc1ncnc(N2CCC(C)(C(F)(F)F)CC2)c1C 20597,C1(C(=O)NCCCC(C)NC(=O)C(c2ccc(F)cc2)=O)CC(=O)NC(=O)N1 20598,O=C(CC1CC12CC2)Nn1cnnc1 20599,N1(C(c2cn(CCC)nn2)=O)CC(CNC(=O)C=Cc2nccn2CC)C(C)C1 20600,C1(NC2(C(N)=O)CCN(C(=O)OC(C)(C)C)CC2)CCC12CCOCC2 20601,N1(C(N2CC(CF)C2)=O)CCC(O)(c2cccc(Br)c2)C1 20602,c1(COC)nc(CC(=O)NCC(=O)N(CCC#N)C)cs1.C(C(C)C)N 20603,C1(C#CC(=O)N2CCC(F)(CNC(c3n[nH]c(C)n3)=O)CC2)(CC)CC1 20604,N1CCc2nccn2CC1.C1(C(O)CCOC(F)(F)F)CCCCC1 20605,C(=O)(C(CNC(C1CCCCO1)=O)CC1CC1)N(CC(CCC)O)C 20606,N1(C(C(CC)NC(C)=O)=O)CCC(C(C)C)CC1NC(=O)CN(CC(C)(C)C)C 20607,C1(NC(C=Cc2n(C)ncc2)=O)CC2(C1)CN(C(C1CC3(C1)CC3(F)F)=O)C2 20608,c1(C(=O)NC(C(C)NC(C2CNC(=O)N2)=O)C)c(F)ccc(O)c1F 20609,N1(C(CC2(C)CC2(Cl)Cl)=O)CCCCC(C2CN(C(C3CCS(=O)(=O)C3)=O)C2)C1 20610,c1(C(=O)NC(CC)CNC(=O)CN(C(C)COC2CCCC2)C)ccccc1 20611,C(C(O)CCNC(c1cc(F)c[nH]1)=O)NC(c1cc(-c2ccccc2)cs1)=O 20612,N1(C(CC2(CC(=O)OC)CC2)=O)CC2CCC(CNC(C3CS(=O)(=O)C3)=O)C2C1 20613,C(CC(=O)NC(C)CCCNC(c1nnn(C)n1)=O)(C1=CCCC1)OCC 20614,C(=O)(C1=C(C#N)CCC1)N1CC(CC(=O)NC2CC(O)C(O)C2)(OC)C1 20615,C1(NC(C2(CC)COC2)=O)CCCC(N(C)C(c2cc(CC(C)(C)C)on2)=O)C1 20616,Cc1cc(NCc2nc(Cc3cccc(F)c3)n[nH]2)n2ncc(Br)c2n1 20617,C1(C(=O)NCCc2ncn(CC)c2)CC(N=[N+]=[N-])CN1C(=O)C(C)NC=O 20618,C(C(CCNC(C1(NC(=O)Cc2ccsn2)CC(O)C1)=O)OC)OC 20619,c1(C(N2CC(N3CCN(C(C4C(C)=C4)=O)CC3)C2)=O)cc2cccc(C)c2s1 20620,c1(CNC(CC2OCCN(C(C(C=C)C)=O)C2)=O)ccc(C#N)cn1 20621,C1(C(N(C2CCN(C(c3cccn3C)=O)C2)CC)=O)CC(=O)N(O)C1 20622,c1(C(=O)NC(C(C)(C)NC(c2ccn(CC)n2)=O)C)c[nH]c2cnccc12 20623,c1(C(N2CC3CCN(c4ncc(C)cn4)C3C2)=O)cccc2ccncc12 20624,N1(C(c2ccsc2Cl)=O)CC2CC(C1)N2C(C1(Br)CC1)=O 20625,n1(CC)cnc2c(N3CC4CC4(CC)C3)nc(N3CCC(CF)CC3)nc12 20626,CCC(C(=O)NC1(CO)CN(C(=O)COOC(F)F)C1)C(F)(F)F 20627,C1(CNC(COCCCC(C)C)=O)CN(c2ccn3nccc3n2)CCC1(C)C 20628,Cc1ccc(CC(=O)O)cc1C(=O)NC1(C(F)F)CCCC1 20629,c1(OCCC#N)ccccc1CNN(C1CC2C=CC1C2)C=O 20630,C(=O)(C=C1SCC(=O)N1C)OC(C(=O)OCCCC)Cc1ccsc1 20631,CC1CC(CO)N1C(=O)C(C1(C)CC1)NC(=O)C(=O)C1CCCC1 20632,S(=O)(=O)(c1cccc(C(F)(F)CF)c1)NCC(C(=O)NC)C 20633,c1(C(C(C)NC(=O)NC(c2cccs2)C)OC)cc(Cl)cc(Cl)c1 20634,Cc1cc(C(=O)NCC(C2CCN(C(=O)C(C)N(C)C)CC2)O)cc(=O)n1C 20635,N1(C(C2C(C)CCCC2)=O)CCC12CN(C(c1nc[nH]n1)=O)C2 20636,C1(C(=O)NCC2(COC)N(C(C(CCCC)C)=O)CCC2)CCc2c[nH]nc2C1 20637,c1(C(N2C(C)(CCC(=O)NC(c3cnc(C)s3)C)CCC2)=O)cc2n(n1)CCO2 20638,CN1CCC2(C(N3CCN(CC(O)C4CC4)CC3)=O)CN(CC(=O)O)CC2C1 20639,C1(NC(c2cc(C(F)(F)F)c[nH]2)=O)CCCN(C(=O)CCCn2cncn2)CC1 20640,N1(C(c2c(C)cccc2)=O)CC2(CC(CNC(=O)CC3(N(C)C)COC3)C2)C1 20641,O=C1CCc2cc(C(N3CC(F)CC3CNC(=O)CCF)=O)ccc2N1 20642,CC1CN(C(=O)C(C)(C)C(F)F)CC1(C)C(=O)NCC(C)(O)CO 20643,CC(C)(C)CC(O)C(=O)NCC1CCCCCN1C(C12CCN(CC1)C2)=O 20644,CC(CC(F)F)C(=O)NCC1(NC(=O)Cc2cc(F)cc(F)c2)CCOC1 20645,n1(C(C)C)cccc1C(c1nnnn1CC1CCCO1)NCCn1ncnn1 20646,C(=O)(C(C)(O)C1CC1)NCCC(C)NC(C1(C2CC2)CC1)=O 20647,N1(C(=O)Cn2cnnc2O)CCN(C(C2CCC23CCOCC3)=O)C2(CCC2)C1 20648,c1(C(N2C(C)CC(NC(=O)C=C3CCN(C)CC3)C2)=O)cc(C2CC2)cc(F)c1 20649,N1(C(C(COC)O)=O)CCN(C(=O)COCc2cccc(C)c2)CC1CCO 20650,c1(CC)onc(C)c1C(=O)NCCC1CC(NC(=O)C(c2cccnc2)C)C1 20651,Cc1c[nH]c2ncc(C(N3CC4CCC3CN4C(=O)CCCC(C)(F)F)=O)cc12 20652,CC(C)CCC(=O)C(=O)NCC1(C)CCCN(C(C2CCCN(C)C2)=O)C1 20653,N1(C(CC(C)n2cc(Br)cn2)=O)CCCN(C(=O)C=CC2CCCO2)CC1 20654,CC(C)CC(C)(C(N)=O)NC(=O)CCCCNC(=O)C(c1ccccc1)C 20655,CC1CC(NC(C2(c3ncccc3F)CCC2)=O)CCN1C(c1ccsc1)=O 20656,N1(C(C(C)OCCCC)=O)CC2(COC)CC1(CNC(=O)Cc1nc[nH]n1)C2 20657,C(CC(CC)C(=O)NC(C1CCN(C(C2(CC)CC2(F)F)=O)CC1)C1CC1)=CC 20658,c1(C(N2C(C)CCC(CC(=O)NCCN(CC)CC)C2)=O)cc2ccncc2[nH]1 20659,CC1CN(C(c2snc(Cl)c2Cl)=O)CC2(CCN(C(=O)CCc3nccs3)C2)O1 20660,c1(CC(C)NC(c2c(CC)csc2)=O)ccc(CNC(=O)C(CC)N(C)C)cc1 20661,C1(NC(CN(CCOC)C(C2CCC(F)(F)C2)=O)=O)CCCC(F)C1 20662,C12(C(=O)NCCCN(C(C)C)Cc3nc(C(C)C)sc3)CCC(C1)C(C)O2 20663,c1(C(N2CC=CC(NC(c3cc(OC)ncc3)=O)C2)=O)ccc(C)c2c1CCC2 20664,c1(CCOC)nc(=NC2CN(C(=O)C(F)(F)C3CC3)CC23CCC3)s[nH]1 20665,C1(CCC)CN(C(c2ccc(OC(C)=O)s2)=O)CCN1C(=O)C(F)=C1CCC1 20666,C1(NC(C(N2CCSCC2)C)=O)COCCN(C(=O)CCCC23CC(C2)C3)C1 20667,O=C(CS(=O)(=O)CCO)NC1CCN(C(=O)Cc2ccc3c(c2)CCC3)C1 20668,CCCC(C)C(=O)NCc1cccnc1.c12cccc(c1)C2.C12CC1NC2=O 20669,N1(C(COCCCOC)=O)CCC(O)(C2(NC(=O)C(C3CC3)SC)CC2)CC1 20670,N1(C(c2c(C)nc(CC(C)C)o2)=O)CCCC(O)(CNC(c2ncoc2C)=O)C1 20671,C1(NC(C(C)CO)=O)CCC2(CC1)CN(C(c1cccnc1O)=O)CCO2 20672,C1(Cl)(C(=O)NC2C(CNC(=O)Cc3cccs3)COC2)CC12CCOCC2 20673,c1(CC(=O)NCCC(C)NC(c2cnc(CCC)s2)=O)csc2ccccc12 20674,C12(C(N)=O)CC(CNC3CCS(=O)(=O)N3)(C1)OC21CN(c2nnc(O)s2)C1 20675,C1(O)(CNCc2c(OC(C)C)cccc2)CCc2ccccc2C1 20676,C(N=c1cc(F)nc[nH]1)C1CCC(NC(C2(C(F)(F)F)CC2)=O)CC1 20677,C12(NC(CCC3CCC(CN)C3)=O)CCC(CC1n1cc(-c3ccsc3)nn1)C2 20678,Cc1cn2c(n1)C(C)CC(C(=O)NC1CC(F)CN(C(c3cnco3)=O)C1)C2 20679,n1(CC)cc(CC(=O)NCCC(C)NC(c2cc(C)oc2C(F)(F)F)=O)c(C)n1 20680,NC12CC(c3nc(C4CC4c4ccccc4)no3)(C1)C2 20681,C(=O)(CCC(CF)CF)NC1CCCC(N(C)C(c2ncn(C)n2)=O)C1 20682,CC(F)(F)C(F)C(=O)NC(C(=O)NCCC1=CCOCC1)c1ccco1 20683,Cc1cc(CN2CCN(C(c3ccnc(Cl)c3)=O)C3CC23)c(C)n1C 20684,c1(COC)csc(C(=O)NC2CCC(N(C(=O)C=Cc3cncs3)C)C2)c1 20685,C#Cc1cc(C2C(C(=O)OC(C)C)C2)ccc1Cl 20686,n1(CC(=O)NC2CC(CCNC(c3c(CC)occ3)=O)C2)c(C)cc(O)cc1=O 20687,C(N=c1nc2c(ncn2C)c(NCc2cn(C)nc2C)[nH]1)C1(S(CC)(=O)=O)CC1 20688,c1(C(N(CC(=O)NCCC(CC)O)C)=O)cnnc(C)c1 20689,CC1=C(C(=O)NCC2(O)CCN(C(C3(CC(C)C)CC3)=O)CC2)SCCO1 20690,N1(C(=O)Nc2c(C(C)=O)cccc2)CC(C)N(C(c2ccccc2)=O)C(C)C1C 20691,N1(C(C(C(C)C)O)=O)CC(C)(C)OC2(C1)CN(C(=O)C=CC=C(Cl)Cl)C2 20692,C#CCCCC(=O)NCC1(C(N2CCC(CCCC=C)C2)=O)CCCO1 20693,c1(CC(=O)NCC2(CC)CC(NC(C3(C#C)CC3)=O)C2)ccc(F)cc1 20694,C1(NC(CC(CC)O)=O)CCCC12CCN(C(C1OCCC1C(C)C)=O)CC2 20695,Cn1nc([N+](=O)[O-])c(Cl)c1C(=O)NCC1C=CCN1C(=O)CCC1CCC(=O)N1 20696,c1(NC(C)=O)cc(C(N2CC(CO)(CNC(=O)C(C#N)C3CC3)C2)=O)ccc1C 20697,c1(C(=O)NCC2C3CN(C(C4N(C)CCCC4)=O)C2C3)ccc2cnoc2c1 20698,C#CCCCCCC(=O)NC1CC(F)(F)CC1NC(=O)C(N1CCCCCC1)C 20699,CC1(C(N2CCN(CC(=O)NCC3(C)CC3(C)C)CC2)=O)CCCCCC1 20700,c1(C(N2CCC(NC(C34CCC(C)(OC3)C4)=O)C2)=O)cnc(O)n(C2CC2)c1=O 20701,N1(C(c2ncc(F)cn2)=O)CC(F)(F)C1C1CC1.C12CC(CO1)C(=O)NC2 20702,C1(CC(=O)NC2C3(CC(OCC)C3)C2)CC2(C1)CN(C(C1CC3CC3C1)=O)C2 20703,c1(NC2CC(=C)C2)cc(N(C)CC2(CCCOC)CC2)nc(COCC)n1 20704,c1(NC(C(N2CCC(C)(O)C2)C2CC=CCC2)=O)ccc(Cl)cc1F 20705,C12(C(N3C(CNC(C4C(C(=O)OC)C4)=O)CCCCC3)=O)CCC(CC1)C2(C)C 20706,c1(NCc2nccc(CC)c2)[nH]c(=NC2CC(NC)C2)nc2c1ncn2C(C)C 20707,C(=O)(C(C#N)C(C)(C)C)N1CCC(NC(c2c(C)ccc(CC)c2)=O)C1C 20708,C(CCSC)(CN=c1cccc(S(=O)(=O)N(C)c2nc3ccccc3s2)[nH]1)OC 20709,Cc1c(C(=O)NC2CC(N(C(=O)CCC3CCCC(O)C3)C)C2)nnn1C(C)C 20710,N1(Cc2cn(C3CCN(C(=O)CC(C4CC4)C4CC4)C3)nn2)CCCCCC1 20711,C(=O)(CC(C)C(C)(C)NC(c1csnn1)=O)NCCn1c(C)ncc1 20712,N1(C(CN2C(=O)CSC2)=O)CCCOC(CNC(=O)CC2CCCOCC2)C1 20713,CC1OC2CCC1(C(=O)NC1CCCC(CN(C(=O)CC3CCCN3C)C)C1)C2 20714,CC(C)CC(=O)NCC1CC1CNC(=O)C(N1CCNC1=O)C 20715,C1(NC(c2c(C)ocn2)=O)CCN(CCCNC(=O)C(c2ccc(C)s2)C)CC1 20716,c1(C(N)=O)ccc2oc(NC(=O)C=Cc3cncc(F)c3)nc2c1 20717,N1(C(C)C)CCCC(NC(=O)C(C)N(C(=O)C(C)(C)CF)C2CC2)C1 20718,CN1CC(C)(C)CC1C(=O)NCC(C(C)(C)C)NC(C1CC2(CC2)C1)=O 20719,N1(C(C(C(=O)OC)C)=O)CC2(CCC(C(=O)Nc3nc(-c4ccco4)cs3)O2)C1 20720,CC(C)CC(C)C(=O)NCC=C1CCN(C(C2(C#N)CCC2)=O)CC1 20721,C1(NC(c2c(C)nc(CNC(=O)CCN=[N+]=[N-])o2)=O)CC(F)(F)C1(C)C 20722,N1(C(C(C)Sc2ccccc2F)=O)CCC(CNC(=O)CCCC(N)=O)C1(C)C 20723,c1(CC)ncc(C(=O)NC2CC(CC(N3CCC3C(C)C)=O)C2)cn1 20724,N1(C(c2cc(C)n(CC)c2C)=O)CCCC2(NC(=O)C(C)CC(N)=O)CC2C1 20725,N1(C(CCC2CCC(C)O2)=O)CCC2(CCN(C(c3cc(CO)[nH]n3)=O)CC2)C1 20726,CC1CN(C(C2CC3(CCC3=O)C2)=O)CCC1NC(=O)CCCC1CCCO1 20727,N1(C(Cn2ccc(C)n2)=O)CCC(O)(C(C)NC(c2ccnc(O)c2)=O)C1 20728,c1(NCC(CCCC)NC(=O)CC(C)CN(C)C)cc(C)nc(OC)n1 20729,C(=O)(CCC(C)CC)NC1CC(CNC(C(CC#C)C2CC2)=O)C1 20730,Cc1ccc(N(C(=O)CN(C)CCc2cccnc2)C(C)C)cc1F 20731,c1(CC(=O)NCCCNC(CC(C)(C)SC)=O)noc2ccc(Br)cc12 20732,C1(NC(Cc2c(C)cccc2)C)CCCCC12CCN(C(=O)OC(C)(C)C)C2 20733,Cn1cccc(C(=O)Nc2ncnc(Cl)c2F)c1=O 20734,CC(Cc1cnn(C)c1)C(=O)N(CCCCNC(=O)C(C)Cc1ccncc1)C 20735,C1(CC(=O)NC(CC)C(C)C)CN(C(c2c(C)noc2N)=O)CCO1 20736,C1(C(N2CC3N(C(CC4CC(=C)C4)=O)CC(C3)C2)=O)COc2ccc(F)cc2C1 20737,C#CCC(C)(CC)C(=O)N1C2CCC(C2)C1CC(=O)NCCC1CCCN(C)C1 20738,N1(CC(=O)NC(C2CCCC2C(=O)OC)C)CC2C(CNC(=O)C3CC3)C2C1 20739,N1(C(c2c(SC)csc2)=O)CC2CCC1C(CNC(=O)C1=C(Cl)CCCC1)C2 20740,c1(C(N2CCC(NC(CS(=O)(=O)NC)=O)C2)=O)c(C)c(C)nn(C)c1=O 20741,Cc1cc(C)c(NC(C2CCCN(Cc3nc[nH]c3C(C)(C)C)C2)=O)c(C)c1 20742,N1(C(c2ccc(CNC(C(CCC)C)=O)s2)=O)CCOCCC1CC 20743,N1(C(c2cc(C)oc2)=O)CC2(CCCN(C(c3ccnc(Cl)c3N)=O)C2)C1 20744,C(=O)(C(C)CC(F)F)NCC(CC)NC(c1ccc(C2(C(F)(F)F)CC2)cc1)=O 20745,c1(C(=O)NCCn2cncn2)cn(CCNC(C2CC2C(F)(F)F)=O)cn1 20746,c1(C(N2CC(CC)C(NC(=O)C3=CCCC3)CC2)=O)cnc2[nH]ccc2n1 20747,C1(CC)CN(C(c2ccsn2)=O)CCC1NC(c1nc(CC)sc1N)=O 20748,CC(C)CC(C(=O)NCC1CCCC1NC(=O)CCc1cnn(C)n1)C(C)C 20749,C1(C(N2C(C(N(C)CC3C(C)C3)=O)CC2)=O)CCCCNC1=O 20750,CCC(C)C(C(=O)NCCC1CN(C(c2sccc2SC)=O)C1)OC 20751,c1(C2CCC(NC(=NC)NCc3ccn(CC)n3)C2)ccc(F)c(F)c1 20752,C1(C(=O)NCC2(CC(=O)NCC3(SC)CC3)CC2)CC(O)C(F)C1 20753,CCC(C)CCCC(=O)NCCC1(NC(c2cn(C3CCC3)nc2C)=O)CCC1 20754,c1(CCC(=O)NCC(C)NC(C(F)CCOC)=O)ccc(OCC(F)(F)F)cc1 20755,C1(N(C(c2c(C)n(C)cn2)=O)C)CCC2CN(C(=O)COC3CC(F)(F)C3)CC12 20756,N1(C(C2N(C)CCN(C(c3scc(C)c3)=O)C2)=O)CCN2C(=O)OCC2C1 20757,CCC(CC(=O)NC1CC(CO)N(C(=O)Cc2cccc(C)c2F)C1)C(C)C 20758,C1(C)(C(=O)NCc2cc(COC)on2)CCN(C(C2CC(=O)CS2)=O)C1 20759,C1(CCC)(NC(=O)COc2cnn(C)c2)CCCN(C(C2(C)CNC(=O)C2)=O)C1 20760,C1(C(=O)NC(CNC(C2(SC)CC2)=O)C(C)C)CCN(c2ccccc2)C1=O 20761,N1(C(c2c(C(C)NC(c3cnn[nH]3)=O)noc2)=O)CCCC12CCNC2=O 20762,Cc1cc(F)ccc1CC(=O)NC1CCCC1NC(=O)CCC1OCCO1 20763,c1(C(=O)NC(C2CN(C(C3(F)CCCC3)=O)C2)C)ccc2c(c1)NC(=O)CN2C 20764,C1(C(=O)OCC)CCC2CCC1N2C(=O)NC1CCN(CC)CC1C 20765,Cc1n[nH]c(C)c1C(C)CC(=O)NCC(C)NC(c1ccc(C(N)=O)[nH]1)=O 20766,N1(C(c2ccc(C)nc2)=O)CCC2CN(C(=O)CN3CCCC3C)C2C1 20767,Cc1ccc(C=CC(=O)NC(C)CC(C)NC(=O)CCc2cccnc2C)nc1 20768,Cc1cc(C2(C(=O)NC3CC3CNC(c3cc(Cl)ccn3)=O)CCC2)cc(C)c1 20769,c1(C(=O)NC2(CCF)C(c3onc(COC)n3)C2)cc(SC)ccc1O 20770,C(=O)(C(C)CCC(C)(C)C)NC1(CC(=O)OC)CC1.CCC1CC(=O)N(C)N1 20771,c1(C(C)C(c2nc(-c3ccc(Br)s3)no2)N)cccc(Cl)c1 20772,CCC(C)(F)C(=O)N1CC2CC2(NC(c2ccc(F)cc2)=O)C1 20773,C1(C(=O)NCCC2(O)CCN(C(C=CCCC)=O)CC2)C2CCC(C2)C1(C)C 20774,N1(C(C(C(C)C)NC(N)=O)=O)CCC(C)C(NC(=O)CCC23CCC(CC2)C3)C1 20775,c1(C(N2CCC(C(O)CO)CC2)C(=O)NCC(=C)C)cc(C)nn1C 20776,C1(C(N2C(CC(=O)NCCC(C)C(F)F)COCC2)=O)CCOC(C)(C)C1 20777,CCCCCC(=O)NCC(=O)NCC1(C)CCN(C(=O)CN(C)CCOC)C1 20778,c1(C(N(C2CCN(C)CC2)CCCOC)=O)cccc(O)c1F 20779,C(CCC[Si](C)(C)C)N(C(Cn1cnnc1)C(=O)O)C 20780,C1(C(=O)NCCCCC2N(C(C3CCC4CC4C3)=O)CCC2)C2CC3C(C2=O)C13 20781,c1(OC)nccc(C(=O)NCC2CCCN(CC3CC4CCC3O4)C2)n1 20782,CCCC(O)(CCC)CC(=O)N(CCNC(C1CCCC1)=O)Cc1ccccc1 20783,c1(C(=O)NCC2C(C)CCN(C(c3cccc(C)c3)=O)C2)cnn2c1NCCC2 20784,c1(CNC(C2CN(C(C)=O)C2)=O)nc2c(s1)CCN(C(=O)CC1COC(=O)C1)C2 20785,c1(C(=O)NCC2C3CN(C(C(CC=C)C)=O)CC32)ccc2c(c1)CC(C)(C)C2 20786,CP(C)(=O)c1cccc(C(=O)NCC2CN(C(C3CCNC(=O)C3)=O)CC2O)c1 20787,c1(CN2CCC(C(=O)Nc3c(OC)cccc3O)C2)c[nH]c2ncccc12 20788,C1(C(=O)NCC2(C(N3CC(C)(OCC)C3)=O)CCCC2)CCN(C)C1C 20789,C12(NC(CCCNC(C3N(CC)CCOC3)=O)=O)CCCN(CCC1)C2 20790,c1(CC(=O)NCC(C)N(C(C(CC)C2CCOCC2)=O)C)ccccc1N 20791,c1(OCC)ccc(C(c2ccccc2C(=O)OC(C)CC)=O)cc1 20792,n1(CC(=O)NCC(CC=C)NC(=O)CC2CC=CCC2)ncn2nccc2c1=O 20793,C1(C(=O)NCC2CC(O)C(O)C2)(CNC(c2csnc2Cl)=O)CC12CCC2 20794,N1(C(C(CC)c2cccnc2)=O)CCCN(C(=O)C=Cc2cnccn2)CC1C 20795,c1(C(N2CCN(C(COCC(=C)C)=O)C(CO)C2)=O)ccsc1S(C)(=O)=O 20796,CN1CC(NC(C2CCOCCN2C(c2cn(C3CC3)nn2)=O)=O)C(F)(F)C1 20797,CN=c1[nH]cc(C(N2CCCC(C3CCCCN3C(=O)CSCC(N)=O)C2)=O)o1 20798,c1(C(=O)NC2C(NC(C(C(C)(C)C)SC)=O)CCCCC2)nc2ncccn2n1 20799,c1(C(N(C)CC2(O)CN(C(CSC)=O)C2)=O)ccn(CC(F)(F)F)c(=O)c1 20800,C1(C(CNC(c2c(C)nsc2)=O)C)CCN(C(=O)C(C)C2(O)CCC2)CC1 20801,C(CCCCC(=O)NC(CCC1CCC1)C(=O)NCc1cccc(C)c1O)OC 20802,c1(OC)ccc(Cn2cc(N(C3COC3)Cn3ccnc3C)nn2)cc1[N+](=O)[O-] 20803,N1(C(CC=CC)=O)CCC(NC(C2CCCC(NC(=O)OC(C)(C)C)C2)=O)CC1 20804,C=C=CCCC(=O)NCCCN(C(=O)CC1(N(C)C)COC1)C 20805,c1(N2CCC(CCOC)C2)nc(C)cc(=NCc2ccc(O)nc2)[nH]1 20806,C#CC1CCCN(C(=O)C(C2CC2)NC(=O)CC2CCCN(C)C2)CC1 20807,C12(C(=O)NC3(CNC(C(C)(C)C)=O)CCCC3)CCCCC1C2 20808,N1(C(C=CCNC(C2CCCC(CF)C2)=O)=O)CCC(O)(CO)CC1 20809,Cc1cc(Cl)c(C(=O)NCC2CC2NC(c2cc3occc3[nH]2)=O)cc1N 20810,N1(CC)CCOC(CNC(=O)CC2CCCN2C(=O)C(C)C2CC2)C1 20811,C(=O)(C(C(C)C)n1cnnc1)N(C1CC1)CC1N(C(C(COC)OC)=O)CCC1 20812,N1(C(C(=O)NC2CCC(SCC(=O)OC(C)(C)C)CC2)=O)CCc2ccccc21 20813,N1(c2nc(C)cc(CC)n2)CC(C2CCCN(C(c3ccsc3OC)=O)C2)C1 20814,N1(C(C2C(C)CC2)=O)Cc2ccccc2C(NC(c2cc(C(N)=O)n(C)n2)=O)C1 20815,C1(NC(c2sc(C)c(O)n2)=O)CC(O)CN(C(C2(C)C(C)(C)C2(C)C)=O)C1 20816,c1(CC)[nH]ccc1C(=O)NC(C1CC=CCC1)C(=O)NCCc1ccco1 20817,c1(CCC(=O)NCCC2(NC(C3CC(=C)C3)=O)CC2)cccc(F)c1 20818,N1(C(C2(COC)COC2)=O)CC(n2cc(CNc3nccs3)nn2)C(O)C1 20819,c1(OC)ccc(NC(=O)CCn2cncn2)cc1.C1C(=O)N1CC(O)C1CCC1 20820,CC1CCN(CC(=O)N(C)CCN(C(=O)COC2CCCCCC2)C(C)C)CC1 20821,c1(C(C2CC2)OC)nc(-c2nc(Cl)oc2C)n(CCC(F)(F)F)n1 20822,C1(NC(CSCC)=O)COC2(CCN(C(c3cc(C)c(C#N)cn3)=O)C2)C1 20823,N1(C(C(C)=C2CC2)=O)CCC(CO)(CNC(C2CCC2(F)F)=O)C1 20824,c1(C(=O)NC(C(C)C)CNC(=O)CC2CCCCCC2)ccc(S(C)(=O)=O)cn1 20825,Cn1cc(C(N2CCc3c(nnn3C)C2)C(=O)NC2CCC2)c(=O)n(C)c1=O 20826,c1(C(N2CC(CNC(c3c(C)cns3)=O)C3(C2)CC3)=O)cc2c(C)cccc2o1 20827,C1(C(N(CCC(=O)N2CC(N3CCC3)C2)C(C)C)=O)C2CCC(=O)C12 20828,C(=O)(CCS(N)(=O)=O)N1C(CN(C(=O)CN2CCCNC2=O)CC)CCCC1 20829,C1(CCNC(C(C)OCC2CC2)=O)CCCN(C(=O)CN2CCS(=O)CC2)CC1 20830,N1(C(COCCC=C)=O)CC2(C1)SCCC2NC(=O)Cc1cccc(Cl)c1OC 20831,C1(CC(=O)N(CC(=O)OC)CC)CN(C(=O)CCCN(C)C(C)C)CC1C 20832,C1(C#N)(C(=O)NC2CC3CC(NC(CC(CC)CC)=O)CC32)CC12CCCC2 20833,C(=O)(CC(C)(C)C)NCc1c(C(=O)NCC(C)C2CC2)nco1 20834,C(C(C)(C)C)N(CC(C1CCC1)NC(CN(N1CCCC1)C)=O)C(=O)C=CCO 20835,C(=O)(C(C)(C)CC(C)(C)C)N1CC2C(NC(CCNC(=O)NC)=O)C(C2)C1 20836,c1(-c2cccc(C=O)c2)c(C)cccc1C.c1(N2N(CC)CC2)ccc(Cl)s1.SC 20837,c1(C(C)NC(c2nc(O)nc(O)c2F)=O)cccc(C2=Cc3ccccc3C2)c1 20838,c1(OCC)c(C(=O)NCCN(C)C(C2(C)CC(O)CN2C)=O)cccc1F 20839,c1(OC)cccnc1C(=O)NCC1COCC1NC(=O)C=Cc1ccc(C)o1 20840,c1(OC)ccc2c(c1)C(C(=O)N(C)CCN(C)C(C1CCC(C)CC1)=O)CC2 20841,c1(Cn2ncc(NC(CC(N3CCC(C)C3)=O)=O)c2)ccc(N)cc1 20842,c1(C(N2CCCC(CN(C(C(C(C)C)F)=O)C)C2)=O)cccc2nc(O)ccc12 20843,CP(C)(=O)c1cncc(C(=O)NC2CCCCO2)c1 20844,CN1CCC(CC(=O)NC2CC(NC(c3conc3C3CCCO3)=O)C2)CC1 20845,C1(CNC(=O)C(N2CCCC(c3nc(O)n[nH]3)C2)=O)CCCC2(CCNCC2)O1 20846,CC(F)(F)C(F)C(=O)N1CCC(C(=O)NCc2cccc(CO)n2)(CF)C1 20847,CCC(C)(CC(NC(=NCCF)NC1CN(c2cccc(C#N)c2)C1)=O)C(N)=O 20848,c1(C(N(C)C)=O)ccc(C(N2CCN(C(=O)CCc3nc[nH]n3)CC2)=O)cc1 20849,c1(C(N(C(CCNC(c2c(C)ccn2C)=O)C)C)=O)ccc2[nH]ccc2n1 20850,c1(CC)noc(CC)c1CC(N1CC(CNC(C2(C)CC3CC3C2)=O)C(C)C1)=O 20851,C1(OC)CCC(CNC(=O)CCCN(C(=O)C(C)Cn2cccn2)C)C1 20852,C1(O)(C(C(=O)Nc2ncn(CC)c2)O)CCOCC1 20853,c1(CC)ccccc1C(=O)N(C(C)C(=O)NCC1CC(C)(C)CO1)C 20854,C1(C(N(CCC(=O)N2CC(N3CCCC3)C2)CC#C)=O)CNC(=O)CC1C 20855,c1(CC)c(C(=O)NC(CNC(C2CC2F)=O)CC(F)(F)F)[nH]c(C)c1C(C)=O 20856,C1(NC(c2ccc(C(F)F)cn2)=O)CCC(C)(C)CC1CNC(C(C=C)(C)C)=O 20857,C1(CNC(C(CC)O)=O)CN(C(c2cnn(CCO)c2)=O)CCCO1 20858,N1(C(C2CN(C(C)C)C2)=O)CCC(CCNC(C2CCSC2)=O)CC1 20859,c1(C(=O)NC(C2CCN(C(C3COC3)=O)CC2)C)ccc2c(F)cc(F)cc2n1 20860,C(=O)(C(Cc1ccccc1)N(C)C)NCC(C)CN(C)C(C1COC(=O)C1)=O 20861,c1(C(N2CC(CC(C)NC(C3CC(=O)N3)=O)C2)=O)coc(C(C)(C)C)n1 20862,C1(CN(C(=O)CC2(O)CCCCC2)CC)CCCCN1C(=O)C#CC1CC1 20863,c1(OC)cccc(OCC(=O)NC(C)C(C)NC(=O)NC2(CF)CCOCC2)c1 20864,CN1CCC(CNC(c2nncs2)=O)C1 20865,N1(C(c2cscc2C)C(=O)NCC=C)CCCCC(CO)C1 20866,Nc1c(C(N2CCC3CCC23CNC(=O)CCC2CCCC2)=O)cccc1Cl 20867,CCC(C#N)C(=O)N1CCC(O)(C(C)NC(C2CCC(C)CC2)=O)C1 20868,C1(C(=O)NCC2C3CN(C(C4CCC45CCC5)=O)CC23)(OC)CCCCCCC1 20869,N1(CC2CCN(c3cc(N)nc4n3ncc4)C2)CC(S(=O)(=O)C2CCOCC2)C1 20870,C1(OC)CN(C(=O)CCNC(=O)C(C(C)C)N(C)C(=O)OC(C)(C)C)CC1CO 20871,C(C)(C(C(=O)NC1CCCC(CC(=O)NCc2cn(CC)nn2)C1)N(C)C)OC 20872,CC#CCCC(=O)NC(C1CCCN(C(C2CN(C)C2)=O)C1)C 20873,C1(N(C(C)=O)CC2CCC(C)(c3cccc(Br)c3)CC2)CCCCC(O)CNCC1 20874,C1(C(N(CCC(C(C)C)NC(=O)CC2CC3CCC2C3)C)=O)CCCCN1N=O 20875,C(=O)(C1=CCC2(COC2)OC1)NCC1C(NC(c2c(C)nccn2)=O)CCC1 20876,C(=O)(C1CCc2cccnc21)N1CC(N(C)C(c2ccc(F)cc2C2CC2)=O)C1 20877,C1(CNC(C=CSC)=O)CCCCC1NC(=O)C(C)OCC(C)C 20878,C1(CCNC(c2cnc(C(C)C)o2)=O)CSCCN1C(c1cccn1C)=O 20879,Cc1cc(C(=O)NCCC2CN(C(C3(Br)CC3(F)F)=O)C2)nn1C 20880,Cc1ccc(C=CC(=O)NCC2CCCN2C(=O)C(C)Cn2ccc(C)n2)cc1 20881,N1(C(C(=O)Nc2cccc(CC)c2)C)CCc2c(ccc(C)c2Br)C1 20882,C12(C(=O)NC3C(NC(C4N(S(C)(=O)=O)CCCC4)=O)CC3)CCC(CC1)CO2 20883,C(=O)(C(=O)CCc1ccccc1)NCC(C(C)C)NC(C1N(C(C)=O)CCC1)=O 20884,N1(C(c2ccc(C)[nH]2)=O)CC=CC(C(N2CCC(O)C2C(C)(C)C)=O)C1 20885,CC(CCC(=O)NCCSCC(=O)NC1(Cl)CC1(F)F)N(C)C 20886,N1(C(C(C)(C)CO)=O)CCC2(CCC2)C(NC(C2CC(F)(F)C2)=O)C1 20887,C1(C(N2CCC(COC)(NC(=O)CCCF)C2)=O)OC(C)(C)OC1(C)C 20888,c1(N2C3CN(C(c4ccc(F)cn4)=O)C(CC3)C2)c(Br)cncc1[N+](=O)[O-] 20889,C1(CNC(CCC=C)=O)CC2(CC2)CN1C(=O)C(C)Cc1cccc(Cl)c1 20890,c1(C(=O)NCCS(CC)(=O)=O)oc(CC2CN(C(=O)C(C3CCOC3)OCC)C2)nc1C 20891,c1(C(=O)NC2C(C)N(C(c3cccnc3S)=O)CC2)ccc2c(c1)COC2 20892,c1(N2CC(CC=C)(NC(c3csc(C(F)(F)F)c3)=O)C2)ccc([N+](=O)[O-])cc1Br 20893,C1(OCC(=O)NCCN(CC(C)O)C(C2(CC)CC2)=O)CCCCC1C 20894,C1(NC(C(C2CC2)OC)=O)CN(c2nc(C)nc(C)c2F)CCC12CCOCC2 20895,c1(NCCCOC(c2ccc3cnnn3c2)=O)ccc([N+](=O)[O-])cc1Cl 20896,C1(N(C=O)Cc2ccc(OCC)c(OC)c2)CCOC2(CCSCC2)C1 20897,C(=O)(C#CC1CCOCC1)N1C(CNC(C(C)OCCN(C)C)=O)CC(O)C1 20898,CCCCCS(=O)(=O)CC(=O)Nc1cc(N2CC(C)OC(C)C2C)ccc1F 20899,C1(C)(N(C)C)CCN(C(C2(CNC(=O)CC3(O)CCCCC3)CC23CCC3)=O)C1 20900,N1(C(C=C(C)C(F)F)=O)CCC(C(CO)NC(=O)Cc2cc(C)cs2)CC1 20901,N1(C(C(=C(C)C2CC2)F)=O)CC(C)CN(C(=O)CC2CCC(F)(F)CC2)CC1C 20902,C1(NC(C2(C)CC=CCO2)=O)CCC12CN(C(c1cccc(C#N)c1)=O)C2 20903,N1(C(C2C(OC)CC2)=O)CCC2(CC2NC(=O)C(C)COC)C1 20904,CC(C)(O)C(F)C(=O)N1CCC(CC(=O)NC2CC23CC(O)C3)CC1 20905,c1(C(C)(C)C)ccc(C(=O)NCC2CC2CNC(=O)C=Cc2ccccn2)cn1 20906,CCC(C)(CN=c1ccc(Br)c(S(=O)(=O)NCc2c(C)cccc2C)[nH]1)C(N)=O 20907,c1(N2CCN(C(c3ccccc3)CC)CC2)nc(C(=O)OC)ncc1F 20908,c1(C(=O)NCC(C2CCOC2)NC(c2scc(C(=O)OC)c2)=O)ncccc1F 20909,C1(C(=O)NCC2C(F)(F)CCN(C(C3CC(=C)C3)=O)C2)CCCCN1S(N)(=O)=O 20910,C1(C(=O)NCC(CC)OC)CC2(CC(NC(=O)C(C3CCCCC3)F)C2)C1 20911,c1(C(=O)Nc2n(CC)nnn2)nc2ccccc2n1CC.C12CCCN(C1)C2=O 20912,c1(CC)cccc(F)c1C(=O)NC1CC(O)CN(C(=O)Cn2cnc(=N)[nH]2)C1 20913,C(C(=O)N1CCC(CCNC(C23CC(F)(C2)C3)=O)C1)(C(C)C)SC 20914,c1(C(N2CC(CNC(c3scc(C)c3C)=O)C3(C2)CC3)=O)snc2ccccc12 20915,Cc1ccc(CC(=O)N(CC(C)NC(=O)C(O)CC2CCCC2)C)c(F)c1 20916,CC1(C)CN(C(=O)Cc2cccnc2Cl)C(CNC(C2(C)CC2C(F)(F)F)=O)CO1 20917,c1(CC)cc(C)c(C(=O)N(C2CCC(NC(c3cn(C)[nH]c3=N)=O)C2)C)o1 20918,c1(C(N2CCC(CC(N3CC(C)C(=O)CC3)=O)CC2)=O)c(F)cccc1C#N 20919,CCCCCC(=O)N1CC(O)CC1C(=O)N(CC(C)(CO)CO)C 20920,Cc1nn(C)c(C(F)(F)F)c1C(=O)NC1CN(C(c2cnccc2Cl)=O)CC1F 20921,Cc1cc(F)cnc1-c1cn(C2CCN2C(c2n[nH]c(O)n2)=O)nn1 20922,C(=O)(CC(C)CC(C)C)NCc1cccc(NC(c2c(OC)n(C)nc2C)=O)c1 20923,c1(CNC(CN(C(=O)C(C)CC2CC2)CC)=O)cncn1C(C)C 20924,c1(C(N(CC(CNC(C2(OC)CCOC2)=O)(C)C)C)=O)ccc(CF)cc1.C(N)=O 20925,C(c1ccccc1Br)=CC(N1CC2C(NC(=O)CN3C(=O)C=CC3=O)C2C1)=O 20926,O=C1CC(C(N2CCC2CNC(C2(O)CCSC2)=O)=O)NC(=O)N1 20927,c1(C(=O)NC(CC(C)NC(C(CCC)OC)=O)C)cnc(C)nc1C 20928,C1(CC=C)(C(N2CCC(C(F)F)C2)=O)CCN(C(=O)COC2CCC2)C1 20929,N1(C(C2CCCN(C(=O)C(O)C3CCC3)C2)=O)CCOCCC1C1CC1 20930,Cc1c(Cl)ccc(C(N2CC(NC(=O)CCC3CCCN3C)C3(CC3)C2)=O)c1O 20931,C1(NC(CCOCCC)=O)CC(C)(C(=O)NCc2cc(C)[nH]n2)C1 20932,c1(C(=O)NC(C(C(=O)NCCCN(CC(C)C)C)C)C)cc(F)ccc1F 20933,C1(CNC(CCn2c(C)ccc2C)=O)CC2(CC(NC(C3CCNC3=O)=O)C2)C1 20934,Cn1cc(C(=O)NC2CCCC(NC(=O)Cc3ccccc3)C2)c(O)nc1=O 20935,Cc1cc(C(=O)NC2CCC2CNC(=O)CNS(N)(=O)=O)cc(F)c1 20936,c1(CC(=O)NC(CNC(c2nc(C(C)=O)sc2)=O)C)ccc(C(F)F)cc1 20937,C1(NC(c2cc(SCC)ncc2)=O)CCCN(C(c2c(N)cccc2F)=O)CC1 20938,c1(C(N(CC(CC)NC(c2oc(C)nc2C(F)(F)F)=O)C)=O)cnc(O)cc1C 20939,c1(CC(=O)NCCCC(C)NC(=O)CCCC(=O)N(C)C)nnc2n1CCOC2 20940,c1(-n2ccc(C(N3CC(c4cn(CCCF)nn4)C3)=O)n2)ccccc1C 20941,C(=O)(C(C)(C)C(C)O)NCC1CC(NC(c2ccc(C(C)=O)cc2)=O)C1 20942,C12(CNC(CCC#C)=O)CC(CN1C(=O)CC1CCCCC1)C2 20943,c1(-c2c(OC)cnc(OC)n2)c(C(F)(F)F)cccc1C1CCc2ccccc21 20944,c1(OC)ncc(C)cc1C(N1CC(N(C(=O)CN2CCCC2C)C)C(O)C1)=O 20945,c1(CC(=O)NCCCNC(c2ccc(F)s2)=O)nsc2ccccc12 20946,c1(C(=O)NCC(CC)NC(C2(C)CC2Br)=O)ncc(C)cc1C(F)(F)F 20947,N1(C(c2n(CCC)ccc2)=O)CCC(C)C1CNC(=O)CCOC1CCC1 20948,c1(C(N(C2CCN(C(C34CC(C(F)(F)F)(CO3)C4)=O)C2)C)=O)cnccc1Cl 20949,N1(C(CCCC(C)C)=O)CCC2(CC1)CC2NC(=O)Cn1nnc2ccccc12 20950,C1(CNC(C(COC)N(C)C)=O)(NC(=O)CC2CCC(=O)N2)CCCCC1 20951,C(=O)(CCCCC1CC1)NCCCN(C(C(C)N(C(C)=O)C)=O)C(C)C 20952,N1(C(CCC#C)=O)CC2CN(C(c3ccc(C#N)c(F)c3)=O)CCC2(CO)C1 20953,n1(C(CC)CC)nc(CCN2CCC(C)CC2)nc1-c1cnc(C(F)(F)F)nc1 20954,CC1(C(=O)NC2CCC(NC(c3ccnc(O)c3)=O)C2)CC2CC2C1 20955,C(C(C)(C)CNC(C12CCC1C2)=O)NC(C1(CC=C)CC1)=O 20956,C(c1ccccn1)=CC(=O)NC1(CC)CN(C(=O)C(C)=C2CC2)C1 20957,c1(C(N2CCCN(C(C(C(C)O)(F)F)=O)CC2)=O)nccc2[nH]ccc12 20958,C(=O)(C1=C(C)C(C)(C)OC1=O)NCC12OCC(NC(C3(CC#C)CCC3)=O)(C1)C2 20959,n1(CC(=O)NC2C3CC(NC(C(C)=C4CCC4)=O)CC32)cccc(O)c1=O 20960,C1(N(C(C(C)OCC)=O)C)CCN(C(c2ccc(-c3ccco3)o2)=O)C1 20961,c1(CN2CC(C(=O)Nc3cccc(OC(F)(F)F)c3)OCC2)cnc(Cl)c(F)c1 20962,c1(CC)ccc(C(=O)NCC2OCCC2C(=O)NCCC(=O)NC2CC2)cn1 20963,c1(NC(c2c(CO)cn(C(C)C)n2)=O)cccc([N+](=O)[O-])c1Cl 20964,C(CCCC(=O)NC(CNC(=O)CCN1CCC(C)CC1)C1CCC1)NC(C)=O 20965,CC1CN2CCN1CC2C(N1CCN(C(c2cc(O)cc(N)c2)=O)C(C)C1)=O 20966,N1(C(C2CC2F)=O)CCC(NC(C2(c3ccc(F)cc3)CCC2)=O)CC1 20967,N1(C(c2c(C)occ2)=O)CCN(C(=O)Cc2ccon2)C(c2ccnn2C)C1 20968,C(N=c1nc(C#N)[nH]cc1Cl)C1C(NC(c2c(C(C)C)ocn2)=O)CCC1 20969,C(=O)(CCCCC(F)(F)F)N1CCC(CNC(C2CCN(CC)C2)=O)C(F)(F)C1 20970,c1(OC)cccc(Cl)c1CC(=O)NC(C)CCNC(c1ccnn1CC#N)=O 20971,N1(C(C(CCOC)C)=O)C2CCC1C(CNC(=O)CSCCC(F)(F)F)C2 20972,C1(NC(C2CC(C)(CC)C2)=O)COC2(C1)CN(C(=O)Cn1c(C)ccc1C)C2 20973,C(=O)(C(CC(F)F)N(C(=O)C(n1ccc(C)n1)C)C)N(CC(C1CC1)OC)C 20974,Cc1cccc([N+](=O)[O-])c1NC(C)CCNC(C1(CF)CCC1)=O 20975,c1(OC)c(C)ccc(C(=O)NCC(CNC(c2cc(C)[nH]n2)=O)OC)c1F 20976,C=CC(C)(CCOC)C(=O)NCC1(CNC(=O)CCCC)CC12CCC2 20977,C(=O)(C(C)CCC(C)(C)C)N1CCCC(CNC(C(C)c2cccs2)=O)C1 20978,c1(-c2cn(-c3ccc(CNC(COCCC)=O)cc3)nn2)ncc(F)cn1 20979,c1(C(n2cc(C(N3CCC(C)(F)C3)=O)nn2)C)c(Cl)cncc1Cl 20980,c1(NCC2(O)CCN(C(Cc3cccc(C)c3F)=O)CC2)cc2nncn2cn1 20981,Cc1ccc(C(=O)NC2CN(C(=O)CSc3n[nH]c(O)n3)C2)c2ccccc12 20982,c1(N(C)C)ncc(C(N2CCCC(CNC(=O)C(F)CC3CCC3)C2)=O)cn1 20983,CC(C(=O)N1CCC(C)(CNC(=O)CCC(C)CN(C)C)CC1)C(F)(F)C(F)F 20984,C(C(C(C)(C)C)NC(=O)CCC(F)F)NC(C(C1CCC(=O)N1)C)=O 20985,N1(C(C(C(CC)C)O)=O)CCC2(CC1)CCN(C(c1ncoc1C)=O)CC2 20986,C1(NC(c2cnn(CC)n2)c2nnnn2CC2CC2)CC2(CCCCC2)C1 20987,N1(C(c2cnc(OCC)nc2)=O)CCN(C(c2nc(C)no2)=O)C2(CC2)C1 20988,c1(C(=O)Nc2scc(C)n2)ccc(OC(F)(F)F)cc1 20989,c1(OC)cc(C(N2CCC(F)(C(=O)Nc3cnc(C(C)(C)C)nc3)C2)=O)nn1C 20990,Cc1cc(CNC(=O)NCc2cnn(C(C)(C)C)c2)on1 20991,C1(C(N(C)C)=O)CCN(C(=O)Nc2csc(C3CCCO3)n2)CC1 20992,c1(CC(C)C(=O)NCC2CN(C(=O)CN(C)C)CC2O)ccc(Br)cc1F 20993,N1(C(CC(C)(C)C2CC2)=O)CCC2(CCCCN(C(=O)CCC3CCCO3)C2)C1 20994,C1(C(=O)NCCCCNC(C2(C)CC(C#N)C2)=O)CCC2(CCOCC2)O1 20995,C1(C(=O)NCC2C(CNC(COCC=C)=O)C2)CCC(C(=O)OC)O1 20996,C1(C)(NC(C2C(C)C2C)=O)CCN(C(=O)CC2CCNC(=O)C2)CC1 20997,C1(NC(c2cc(CCCCC)[nH]n2)=O)CCC2CN(C(C)C(=O)NC)CC2C1 20998,c1(N(C(C)=O)C)ccccc1C(=O)NCC1CC1NC(=O)CCc1ccon1 20999,C=CCCN=C(NCCc1ncc(C)cc1C)NCC1CN(C(=O)OC)C1 21000,CCCCCCCCC(=O)N1CCN(C)C(CNC(C2C3CCC(F)(F)C23)=O)C1 21001,C1(C(N2CCC(N(C)C)C2)=O)CC2C=CC1N(C(=O)C(C)(C)C(=O)N(C)C)C2 21002,Cc1cc(Cl)c2ccc(C(N3CCC(C(C)NC(=O)CC(C)C)CC3)=O)cc2n1 21003,C(=O)(CCC1CCc2ccccc21)N1CCC(CNC(CCCCC)=O)C1 21004,C(=O)(C1CC(=O)c2c(F)cccc21)N1C2CN(C(C3CCC(=O)N3)=O)C(CC2)C1 21005,c1(C(N(CC(C)NC(=O)C(F)n2ccnc2)C)=O)cccnc1N(C)C 21006,C(=O)(CC(C1CC1)NC(=O)CCCn1cnnn1)NCCC=CC=C 21007,C=C(C)CCC(=O)N1CC(N2CCN(C(=O)Cn3ccc(C(=O)OC)n3)CC2)C1 21008,CCC(C(=O)NCC1CN(C(c2nnn(C(C)(C)C)n2)=O)C(C)(C)C1)C(C)(F)F 21009,C(CC(C)C(F)(F)F)NC(c1n(C(C)(C)C)nnn1)CCC1OCCO1 21010,C1(NC(=O)NC(C2CCCN(CC(N3CCNC(=O)C3)=O)C2)C)CC(=O)NC(=O)N1 21011,c1(C(=O)NC(c2cn(C)nn2)C)cccnc1CNC(C1CC2CCC1C2)=O 21012,N1(C(C(C)(C)NS(C)(=O)=O)=O)CCC(NC(=O)CC2CCOC2)C1C1CC1 21013,N1(C(CCc2c(C)noc2)=O)CCC(C)(C)C1CNC(c1cc(F)cc(F)c1)=O 21014,c1(NC(=O)NC2CCN3CCCC3C2)ccn2c(O)nnc2c1 21015,c1(CC(N2CCC(NC(COC(CC)CC)=O)C2CC)=O)cc(F)ccc1C 21016,CC1CN(C(=O)CN2CCCC2)CCC1NC(C1(C2CC2)CC1)=O 21017,CC1(C)CCC(O)(C(=O)NCC(O)CNC(C2CCC=CO2)=O)CC1 21018,N1(C(Cc2c(C)ocn2)=O)CCC2(CC1)CC(C)N(C(=O)CCS(C)(=O)=O)C2 21019,c1(COC)ncc(C(=O)NC(C)(C)C(C)NC(C2C(C)C2C)=O)c(=N)[nH]1 21020,c1(CC(=O)NC2(C)CCN(C(C(CC)F)=O)C2)nn(C)c(=O)c2ccccc12 21021,c1(NC(C(C)NC(C)=O)=O)cn(C)nn1.C1(CC)CCN(C(=O)CCC2CC2)C1 21022,C1(CNC(C2CC(C(C)(C)C)C2)=O)CCCCCN1C(C1CC12CC2)=O 21023,c1(C(=O)NCCC(C)N(C)C(C2CC(O)C2)=O)c[nH]c2cc(Br)ccc12 21024,c1(N(C(C)CCNC(C2CCCC(O)C2)=O)C)snc(Cl)c1C#N 21025,Cc1nncc(C(N2CC3CCC3(CCNC(c3cnsn3)=O)C2)=O)c1C 21026,c1(C(=O)NCCN(CC(C)O)C(C2CC23CC3)=O)cn2ccnc2s1 21027,C(C)(C)(CCC(=O)N1CCCC(NC(c2nn(C)nc2Br)=O)C1)OC 21028,C#CC1(O)CC(C(=O)Nc2cccc(NC(=O)C(COC)CC)c2)C1 21029,CCCCCC(C(=O)N(CCCN(C(=O)CN1CCCCC1C)C)C)C(C)C 21030,c1(C(C(N2CC(C)C(NC(=O)C3=CCCC3C)C2)=O)=O)ccc(F)cc1F 21031,c1(C(=O)OC)ccc(F)c(-c2cnc(SC)s2)c1OC 21032,c1(CC(C(N2CC(CCO)(NC(Cc3nc(C)[nH]n3)=O)C2)=O)C)ccccc1C 21033,c1(C(N(C)CC2(CNC(C3(O)CCOC3)=O)CC2)=O)ccc(C2=CCCC2)cc1 21034,C1(NC(c2c(CC)cno2)=O)CCC2(CC1)CN(c1nnc(C3CC3)s1)C2 21035,N1(C(=O)CCC2CCOC2)CC2CCC1CN2C(c1cc(C(F)F)cs1)=O 21036,c1(C2(C(N3CC(CNC(CC=CC)=O)C(N(C)C)C3)=O)CC2)ccc(Cl)cc1F 21037,C(CCOC)(C(=O)NCCN(C)CC)NC(C(C=C)N(C)C)=O.C(COC)S 21038,c1(N2CCCC(CCNC(C3OCC(C)C3)=O)C2)nc(C2CC2)nc(=N)[nH]1 21039,C1(C(N2CCN(C(c3nc(CC)sc3)=O)CC2CF)=O)CCc2ccnn2C1 21040,Cc1ccc2c(c1)c(CCNC(c1cc3c(Br)cnn3cn1)=O)cn2C 21041,C(=O)(C1CCc2ccccc21)NC1CC2(CN(C(C3=CCCN(C(C)=O)C3)=O)C2)C1 21042,C(CS(=O)(=O)CC(=O)NCC1CCCC1NC(=O)C=Cc1ccoc1)OC 21043,C1(C(=O)NCC#CC)C=CC(NC(=O)CC(=O)OCC)C1 21044,c1(C(C)=O)cc(C(=O)NCC2(C)CCCN2C(c2cccnc2C)=O)n(C)c1 21045,FC1CCCCCC1N=c1[nH]c(=NCC2CC3(CCOCC3)CO2)[nH]c2c1SCC2 21046,N1(C(=O)OCC)CCC(CC(=O)NC(CNC(=O)CCCC2CCC2)C(C)C)C1 21047,C1(OCc2cc(C)on2)C(C)CN(C(=O)C(=O)NCC(=O)N)CC1C.C(C)(C)(C)O 21048,C=CCN=C(NCc1cnn(Cc2ccccc2)c1)NC1CC12CCC2 21049,N1(C(C(C)C)=O)CCC(NC(c2ccon2)=O)C1c1ccccc1 21050,CC1Cc2cc(CC(N3CCCC(CNC(=O)C=C4CCC4)CC3)=O)ccc2O1 21051,C1(C(=O)NCC2(OC)CN(C(=O)C(C)N3CCCC3)C2)CC2(CCO1)CC2 21052,Cc1nn(C)c(C(=O)NC2CC(NC(=O)CCNC(=O)C(C)(C)C)C2)c1[N+](=O)[O-] 21053,C1(NC(c2occ(C)c2)=O)CCCCC1NC(C1CCC(C(N)=O)O1)=O 21054,c1(OC)ccc2nc(C(=O)N(CCC#N)CCNC(=O)CNC=O)ccc2c1 21055,C1(NC(C2CC(C(C)C)C2)=O)COC2(C1)CN(C(c1coc(C(N)=O)c1)=O)C2 21056,N1(C(C2N(C(C)=O)CC(O)C2)=O)CC2(CC(NC(c3cccc(F)c3O)=O)C2)C1 21057,CCCCC(CCCC)NC(C1CC(F)CCN1C(C1CCCC(=O)N1)=O)=O 21058,CC1(C)CCCC1C1CCN(C(N2CCCC3CC(O)CCC23)=O)C1 21059,C1(CNC(C(COC)C)=O)CC(NC(c2ccc(C(=O)OC)cc2)=O)C(O)C1 21060,c1(CC(=O)NC2CCCC(c3cccc(Cl)c3)C2)cc(Cl)ccc1I 21061,c1(OCC)ccc(C(=O)NC(C)CCCNC(c2nccc(C(F)F)n2)=O)cn1 21062,C1(NC(=O)C(F)C2CCC2)CCCCN(C(c2cnc(C(F)F)cn2)=O)C1 21063,CC1(F)CC(C(=O)NCCC2(O)CN(C(c3cnoc3C3CCOCC3)=O)C2)C1 21064,C(N=c1nc(N2CCCNC(=O)C2)c2ncccc2[nH]1)c1ccc(C)cc1N 21065,C1(C(=O)NC2CC(CC)OCC2)CCN(C(c2cn(C)nn2)=O)C12CC2 21066,c1(OC)nc(N2CCCC2CNC(=O)C(F)(F)c2ccccc2)cc(C)n1 21067,CC1(C)NC(=O)CCC1NC(C1CNC(=O)CN1C(=O)CP(C)(C)=O)=O 21068,c1(OC)cc(F)c(C(=O)NCCC(C)NC(=O)CC2C(=O)N(C)N=C2C)c(Cl)c1 21069,c1(C(C)C)nc2ccccc2nc1SC1CCN(C)CC1 21070,c1(OC)cc(F)c(Cl)cc1C(N1CCC(NC(C2CN3CCN2C(C)C3)=O)C1)=O 21071,C1(C2CCN(C(=O)C3=CCCSC3)CC2)(NC(C(C)NS(C)(=O)=O)=O)CC1 21072,c1(OC)ccc(F)cc1NC(C1CC1C(=O)Nc1ccc(Br)c(F)c1)=O 21073,C#CCC(CC(=O)N1CC(n2cccn2)C1)NC(=O)CCNC(=O)COC 21074,c1(C(=O)NCC(CNC(CCc2ccc(C)s2)=O)O)ccccc1OCC(C)C 21075,c1(OCC)cccc(C(=O)NC(C2CCN(C(=O)Cc3conc3C)CC2)C)c1 21076,c1(C(=O)NC2(COC)CN(C(=O)Cc3ccsc3C)C2)cnc2c[nH]nc2c1 21077,CC(CC(=O)N1CC(C)(C)CC1CNC(C1CCc2ncnn2C1)=O)C(F)(F)F 21078,C1(NC(C2CC(O)CN2C(=O)CCN2CCC(F)C2)=O)CCCN(O)C1=O 21079,c1(C(N2CCC(F)(CNC(C3CCC3F)=O)CC2)=O)ccc2c(c1)CNC2=O 21080,N#Cc1ccc(C(N2CCCC(NC(=O)C=CC3CCOCC3)C2)=O)nc1 21081,N1(C(CN(CC(C)C)C(c2cn[nH]c2)=O)=O)CC(CO)OCC1C 21082,C(CCCCCCCO)=CC(N1C(CCNC(CCCC#C)=O)CSCC1)=O 21083,N1(C(C2CCN(C(C)C)CC2)=O)CC(O)C(O)C1CNC(=O)CCCCCO 21084,C1(NC(C(CC)NC(C)=O)=O)CN(CC2(c3ccc(F)cn3)CC2)CCC1CO 21085,CCC(C)CC(=O)N1CCCC1CN(C(=O)CCCCc1ccccc1)CC1CC1 21086,C(=O)(CC(O)c1ccccc1)NC1C(NC(C(F)=CCC)=O)CC1 21087,CC1CCC(F)(C(=O)NCC2(C)CCCN2C(c2ccc(CCF)cc2)=O)CC1 21088,Cc1cc(OCCCN2CCCC2)ccc1N1CCCC1=O 21089,C=CCC(C)(C)CCNC(=O)C(C)(C)Cc1cn(CC=CCC2CCOCC2NC)nn1 21090,N1(C(c2c(CCC)nns2)=O)CCN(C(c2ccc(C(C)F)cc2)=O)CC1CC 21091,C(=O)(C1CCCn2cncc21)NCC(CNC(c1sc(C)c(O)n1)=O)(C)C 21092,C(=O)(C(O)CC(F)F)N1CCC(O)(CNC(c2c(CCC)n[nH]c2)=O)C1 21093,S(=O)(=O)(c1cccc(N2CCCC(CCO)CC2)n1)NCC(CC)C(C)C 21094,C1(C(=O)NCC(N(C)C(C2CC(F)C2)=O)C2CC2)CCOC(C)(C)C1 21095,N1(C(CCNC(=O)OC)=O)CCN(C(=O)C=CBr)C(CO)C1 21096,C(=O)(C(C)(C)C(=O)NC(c1cccc(OC)c1)CNC(=O)C1=C(Cl)CCC1)OC 21097,C1(C(N2CCC(C(CNC(=O)CCc3cn[nH]c3)F)CC2)=O)CCC(F)(F)CC1 21098,c1(NCC2CCCN(C(C3(CC#C)CCCCO3)=O)C2)cc(C)nc2ncnn12 21099,n1(C(C)C)ncnc1CNC(=O)C=CC(c1cnn(C)c1)=O 21100,N1(C(C2CN(S(CC)(=O)=O)C2)=O)CC2CCCC2(NC(=O)CCC2(C)CC2)C1 21101,CC1=C(C(=O)N(C2CCCC(NC(c3c[nH]nc3C3CCC3)=O)C2)C)CCO1 21102,CC(C)CCCC(=O)NC1(CF)CCN(C(c2coc3c2CSC3)=O)C1 21103,CC(C(=O)N1CC2(CC2)CC1CNC(=O)C(c1ccccc1)C1CC1)C(C)(F)F 21104,C(=O)(C(C)(CC)C(=O)NC(C)CCNC(=O)CNC(=O)CC(C)(C)C)OCC 21105,C1(CNC(c2[nH]cc(CC)c2)=O)CN(C(c2n[nH]c(C(C)(C)C)n2)=O)CCN1C 21106,C(=O)(CCCCCCS(N)(=O)=O)NC(c1cn[nH]c1)CNC(C(C)OCC)=O 21107,C1(C(N2CC(OC)C(C(N3CCC(N(C)C)C3C)=O)C2)=O)CCC2(CC1)CC2 21108,c1(C(N(C2CCN(C(=O)CC=CC(C)(C)C)C2)CC)=O)n[nH]c2c1CCC2 21109,C#CCC(O)C(=O)N(C)CC1CCCCN1C(=O)CCSCc1ccc(C)cc1 21110,S(C(F)(F)F)CC(=O)NC1CC(N(C(CNC(C)=O)=O)C)C1 21111,c1(OC)c(CN=C(NCC(=O)NCC2CCOC2)NC2CC2(F)F)cccc1F 21112,N(C1CC(C)Sc2ccccc21)C(=O)Nc1cc2nc(CC(C)(C)C)oc2cc1 21113,C(CC(N)=O)(C(=O)NCCN(C)C(c1cc(C(C)C)on1)=O)NC(CC(C)C)=O 21114,C1(O)(CCNC(C(C)Oc2cccnc2)=O)CCN(C(c2nc(=N)cc[nH]2)=O)C1 21115,c1(C(=O)OC)ncccc1NC(=O)CNc1[nH]c(C)nc1Cl 21116,C1(C(=O)NCCCC)CCCN(C(c2cn(CC)nn2)=O)C1CC 21117,C1(CCNC(C=COCC)=O)CN(C(=O)C(C)CNC(=O)OC(C)(C)C)CCO1 21118,c1(C(N2CC(C#N)(CF)C2)=O)nc2ccccc2s1.C12CCN1C2=O 21119,N1(C(C=C2CCC(C)CC2)=O)CC2CC(C(=O)NCCC#CCO)(C2)C1 21120,c1(C(CC(=O)NCCCNC(c2cn(CCOC)nn2)=O)C)ccc(F)cc1F 21121,C1(C(N)=O)CN(C(c2csc(C(N)=O)n2)=O)CCC1NC(C1(C)CCC(=O)C1)=O 21122,c1(C(N2CCC(F)(C(=O)OC(C)(C)C)CC2)=O)cc2n(n1)CCCN2 21123,Cn1nc(C2CC2)cc1C(=O)NC(C1CCOC1)CNC(C1CC(O)C1)=O 21124,c1(CNC(C)=O)cc(C(=O)NC(COC)CO)c2n1CCOC2 21125,N1(C(CCSCC)=O)CCC(C2CCC2)(CNC(c2cc(=O)n(C)o2)=O)CC1 21126,CC(C)C(C(=O)N(CCCCN1CCCC1)C)NC(=O)C(C)Oc1ccccc1 21127,CN1CCCC(O)(CC(=O)NCCN(C(=O)CC(F)(F)F)CC2CC2)C1 21128,c1(CC(=O)NCCCC2CN(C(c3c[nH]ccc3=O)=O)CCO2)ncncc1Cl 21129,Cc1ccc(F)cc1-c1ccc(NC(=O)NC(C)(C(N)=O)C(C)C)cc1 21130,CC(C)C(C(=O)NC1(CNC(=O)CSc2cccc(Cl)c2)CC1)c1ccn(C)n1 21131,CC(C)CC(O)C(=O)NC1CCN(C(=O)CN2CCN(C)CC2)C1C(C)(C)C 21132,C1(CNC(c2ccc(CC)o2)=O)CC2COCC2N1C(c1c[nH]c(C)cc1=O)=O 21133,N1(C(C)=O)CCC(NC(=O)C(C(C)C)NC(C2CCCC2)=O)CC1 21134,C1(NC(C(C)NS(C)(=O)=O)=O)C=CCN(C(c2cc(-c3ccoc3)on2)=O)C1 21135,N1(C(C(CC#C)O)=O)CCn2nc(CNC(C3(O)CCCC(C)(C)C3)=O)cc2C1 21136,C1(NC2CC(C(F)(F)F)(OC)C2)CNC2(CCC2)C1 21137,N1(C(C2CCN(C(C)=O)CC2)=O)CC(C)CN(C(=O)COc2ccsn2)CC1C 21138,Cn1c(C(=O)NC2CCCN(C(c3ccc(S(C)(=O)=O)s3)=O)C2)ccc1[N+](=O)[O-] 21139,N1(C(C(C)CF)=O)CCC(C(C)(C)CNC(C2(O)CC(C)(C)C2)=O)CC1 21140,C1(NC(c2c(OC)nsc2)=O)CC(C(=O)NC2CCNC(=O)C2)C1(C)C 21141,C1(O)(CNC(C(C=C)(F)F)=O)CCCN(C(C2CCN(C(N)=O)CC2)=O)C1 21142,c1(NC(=O)Nc2ocnc2-c2cn(CC3CCCOC3)nn2)ncc(Br)cc1F 21143,CC1CCCCC1CN1CCC(NC(=O)CNC(=O)NC2CCOCC2)CC1 21144,CC1CCN(C2CCNC2)C(NC(=O)CSc2nnnn2-c2ccccc2)C1 21145,c1(C(=O)NC2(CNC(c3ncccc3Cl)=O)CC2)c(O)nnc2c1COCC2 21146,C1(CCC)(C(=O)NC(C)CNC(C2CCC2n2ccnc2)=O)CCC1 21147,C(CNC(=O)CCCC1(NC(c2ccc(CO)o2)=O)CCC1)(C(F)(F)F)OC 21148,Cc1sc(O)nc1C(=O)NCC(C12CCC(CC1)C2)NC(C1CCC(O)C1)=O 21149,c1(C(C(=O)NCCCCCNC(C=C(CC)C)=O)C)cccc([N+](=O)[O-])c1 21150,CCCCCCCC(=O)NCC1(F)CC(NC(=O)CCc2cnco2)C1 21151,C(CC(C(=O)N1CC(COC)C1)NC(C1CCNC1=O)=O)=CC 21152,N1(NC(C23CC(Nc4cnccn4)(C2)C3)=O)CCN(Cc2ccnc(Cl)c2)CC1 21153,c1(OCC)ncc(C(=O)NCCC(O)CNC(=O)CCC2CCCOC2)s1 21154,N1(C(C(n2c(C)ccn2)C)=O)CCC(C2CCCN2C(=O)C(O)CN(C)C)CC1 21155,CCS(=O)(=O)CC(=O)NC1CCN(C(=O)CSc2ccc(OC)cc2)CC1C 21156,C1(C(=O)NCC(C)NC(=O)COCC2CCOCC2)Cc2ccccc2S1 21157,c1(C(=O)NCc2ccsc2-n2cnnn2)ncsc1-c1ccccn1 21158,C(=O)(C1CCCc2scnc21)NC1C2N(C(c3ncc(C)cc3F)=O)C(CC2)C1 21159,C(=O)(CC(O)CC(C)C)N1CC(n2cc(CCCC)nn2)C(O)C1 21160,N1(C(CC2(O)CN(Cc3ccc(CC)o3)C2)=O)CCCC(CN2CCCC2)C1 21161,CC1(C)NC(=O)OC12CCN(C(=O)C(C1(O)CCCCC1)(C)C)C2 21162,N1(C(c2cncc(C)c2C)=O)CCC2CN(C(=O)C(O)C3CC3)CC12 21163,c1(-c2c(C)ccc(C(F)(F)F)c2)ccc2[nH]c(C(N3CCNC(=O)C3)=O)nc2c1 21164,C1(CC(=O)NCC(c2cc(F)cc(Cl)c2)NC(C(C)=CC)=O)CC2CCC1CC2 21165,N1(C(CCc2ccc(C)o2)=O)CCOCC1CNC(c1ncoc1C(C)C)=O 21166,CCC(CC(=O)N1CCC(NC(=O)Cc2ccon2)C(O)C1)C(C)C 21167,C12(CNC(C(C)OCC=C)=O)CC(NC(=O)C=Cc3ccncn3)(CO1)C2 21168,N1(C(C2C(C(C)=O)C2)=O)CC(CNC(c2ccc(=O)n(CCO)c2)=O)CC(C)(C)C1 21169,C1(CC(=O)NCC2CC2c2ccc(Cl)cc2)CCN(C(C2(CO)CCC2)=O)CC1 21170,c1(C(=O)NCC2C(CNC(C3CCC(N(C)C)CC3)=O)C2)ccn2cnnc2c1 21171,c1(CC)ccc(C=CC(N2CCN(CCNC(C3CCCC3C)=O)CC2)=O)cc1 21172,N1(C(=O)CCCCc2cn(C3(C(=O)O)CC3)nn2)CCCN(c2nncs2)CC1 21173,C1(CNC(C2(C)CC2)=O)CN(C(=O)COc2ccc(CC#N)cc2)C2(CCC2)C1 21174,c1(CC(N2CC(NC(CC(C(=O)OC)C)=O)C(C)(C)C2)=O)ccn2cncc2c1 21175,CN1CCOC2CN(C(=O)C3=CCN(C(C4CCOCC4(C)C)=O)C3)CC12 21176,C=CC1CCC1C(=O)N(C1CN(C(=O)C=CC(CC)=CC)C1)C 21177,c1(C(=O)NCCN(C(c2oc3ccccc3c2Cl)=O)CC)ccc2nncn2c1 21178,Cc1noc(C)c1CSCC(N1CC(NC(c2cc(C3CC3)no2)=O)C(C)C1)=O 21179,c1(C(N2CC(C(N3CCC(F)(CO)C3)=O)CC(C)C2)=O)ccc([N+](=O)[O-])cc1O 21180,c1(C(C(=O)NC2CCCC2)N(CC(COC)C)C)ccncc1F 21181,N1(C(C)C(=O)NC23CC(CNC(=O)COCC4CCC4)(C2)C3)CCN(C)CC1 21182,c1(C(C)O)ccc(C(=O)NCC2CCCCN2C(=O)C(F)=CC2CC2)cc1 21183,C(=O)(CCCC(=O)NCC(CO)NC(c1cccc(C2CCC2)c1)=O)N(C)C 21184,N1(C(CN(C)C)=O)CC2CCC(CNC(=O)C(C)(F)c3ccon3)C2C1 21185,C1(CNC(c2cscn2)=O)CN(C(c2ccc(F)cc2F)=O)C2CCN1C2 21186,Cn1cnnc1CCCC(=O)NCC1C=CCN1C(c1cnc(C(F)F)s1)=O 21187,C(C(=O)Nn1cccn1)C1C(C)CCC1.C12(CCCCC1)C(=O)N2 21188,C1(CCC)(NC(=O)Cc2ccc(OC)c(Cl)c2)CCN(C(=O)C2=COCC2)CC1 21189,c1(CC)n[nH]cc1CNC(=O)C=CC(C)(C)NC(=O)C(F)=C(C)C 21190,C1(O)(CNC(C2CC3C=CC2C3)=O)CCN(C(c2ccn(CC(F)F)n2)=O)CC1 21191,C(CC(C)C(F)(F)F)NC(C(C1(O)CN(C(C2(COC)CCCO2)=O)C1)F)=O 21192,C1(C(=O)NCCC(C)N(C)C(c2cc(O)nc(Cl)c2)=O)CC1C1(C)CCOCC1 21193,C(C(CC(C)C)C(=O)NC1(C(=O)NCC#CC(F)(F)F)CC1C)OC 21194,c1(C(=O)NC2CC3(C(NC(c4c(C)onc4)=O)C3)C2)cc2c(o1)CCCC2 21195,C1(NC(=O)NCC(CSC)(C)C)CCC2(CC1)CC2C#N 21196,C1(COC)(CNC(C2CCC2(C)C)=O)CCN(C(c2cc(Cl)nnc2O)=O)CC1 21197,C(CC(F)F)(C(=O)N=c1ccn(C(F)F)[nH]1)N(C(C(COC(C)=O)C)=O)C 21198,c1(C(CNC(CC2(N)CC2)=O)F)cccc(Br)c1 21199,c1(C(N2CC3C(CNCc4cncc(NC)c4)(C3)C2)=O)cc(OC)c(O)c(Cl)c1 21200,C1(NC(C2CN(CCOC)C(=O)C2)=O)CN(C(C2(C)CCCCC2)=O)CC12CC2 21201,C1(NC(C2C(NC(C(=O)N(C)C)=O)C2)=O)CCCC1C(C)(C)C 21202,c1(C(=O)NC2COCCN(C(C(COC)(C)C)=O)C2)ccc2ccccc2c1F 21203,Cc1ccnc(C(=O)NC2CCC(C(=O)NCC(c3ccccc3)O)C2)c1 21204,N1(C(c2ccc(C)cc2C)=O)C(C)CC2CN(C(=O)C(C)C(O)C(C)C)CC12 21205,C1(c2cccs2)(C(=O)NC2C(CNC(C(C=CC)O)=O)C2)CCCCC1 21206,c1(C(N2CCC3(CC2)CC(=O)N3)C(=O)NCC=C)ccc(C)c2c1CCC2 21207,N1(C(C(CC)OC)=O)CC2CCC(NC(c3cnoc3C)=O)CC2C1 21208,CS(=O)(=O)C1CN(C(C2CCOC2)=O)CC1NC(c1cn2cc[nH]c(=O)c2n1)=O 21209,N1(C(CCN(CC=C)C(C2CC2F)=O)=O)CCC2(CCCO2)CC1 21210,C(=O)(CCC(C)(C)NC(=O)CCCC1CC1)N(CCOC)CCF 21211,c1(C(COC)NC(C2CC(O)(CO)C2)=O)ccc(F)cc1 21212,c1(SCC)cnccc1C(=O)NCCC(C(C)C)NC(=O)C=CC1CCCN1C 21213,Cc1cc(C)c(CC(=O)NC2C=CCN(C(c3n[nH]cc3C)=O)C2)c(C)c1 21214,C1(NC(CNC(=O)OC)=O)C2CC1CN(C(=O)NC1(C(F)(F)F)CCC1)C2 21215,N1(C(c2ccn(C)n2)=O)CC(CNC(=O)COc2ccccc2)C2CC12 21216,N1(C(c2c(CN(C)C)ccs2)=O)CCC(C)(NC(c2cnncc2O)=O)C1 21217,CC12CC(NC(C3CCC3(C)C)=O)(C1)C1(CCN(c3ncnc(Cl)c3Br)CC1)O2 21218,c1(C(=O)NC(C)CNC(=O)C(F)(F)c2csc(Cl)c2)cnc(N)cn1 21219,N1(C(c2cccc(CC=C)c2)=O)CC(C)C(NC(=O)CNS(=O)(=O)NC)C(C)C1 21220,CCC(C)(CCC(=O)OC)NC(c1cc(CCN)on1)=O 21221,C1(O)(CC(=O)NCc2ccc[nH]2)CN(C(c2ccsc2)=O)C1 21222,N1(C(CCC)C(=O)NCCCC(=O)OCC)CC(C)CCC12CC2 21223,C(=O)(C1CCCc2nnn(C)c21)NC(CNC(CCCCC)=O)CC(F)(F)F 21224,CCCCC(O)C(=O)N1CCC(C)(NC(=O)CC2CCCNC(=O)C2)C1 21225,C1(NC(c2cc(COC)[nH]n2)=O)CC(C(=O)NC2CCNC(=O)C2)C1(C)C 21226,C1(CC)CN(C(C2CC(C)(N)C2)=O)CC(C)S1=O 21227,N1(C(C(=O)N(C2C(CC(C)C)OCCC2)CC(F)F)=O)CCc2ccsc2C1 21228,c1(C(=O)NC2CCN(C(C(CC)NC(N)=O)=O)C2(C)C)ccc2c(n1)CCCN2 21229,C12(C(=O)NC(c3ccc(N4CCOC4=O)cc3)C)CC(C1)C(C(F)(F)F)N2 21230,CCCC(CC)CCC(=O)NC1CN(C(C2(N(C)C)CCC2)=O)CC(F)(F)C1 21231,Cc1ccc2c(c1)CC(NC(c1occc1-c1ccc(F)c(F)c1)=O)C2 21232,C(=O)(CC(C)CC(F)(F)F)N(C1CCN(C(=O)C=C2CCC2)C1)CC#C 21233,N1(C(C2CC(C)C2)=O)CCOC2CCN(C(=O)Cn3cnc([N+](=O)[O-])c3)CC12 21234,N1(C(c2c(COCC)nn[nH]2)=O)CC2CC1CN2C(C1CC1OC(C)(C)C)=O 21235,C(C(=O)N1CCC(C)(NC(=O)C(F)=CCCF)CC1)(C(C)(C)C)SC 21236,N1(CCCNC(c2c(C)occ2)=O)CC(NC(c2coc(O)n2)=O)CCC1C 21237,N1(C(C(CN(C)C)(C)C)=O)CC2(CCC(CNC(=O)CSCc3cscn3)O2)C1 21238,c1(C(N2C(C(C)NC(CCSCCCC)=O)CCC2)=O)cn(C)nc1OC 21239,C(CC(C)(C)C(=O)NCC1(F)CN(C(=O)CCCCCN(C)C)C1)SC 21240,c1(C(N2CCN(C(c3ccc(CC)s3)=O)CC2CF)=O)ccc2cccnc2c1 21241,c1(C(N2CC(C)(NC(C3C(SC)CCC3)=O)C2)=O)nn(C)c(C(F)(F)F)c1Cl 21242,C1(C(N(C)Cc2cccc(NC(=N)N)c2)=O)CCCN(c2cnn(C)c2)C1=O 21243,C1(CC(=O)N(CCCC)CC)CN(C(=O)C(CN(C)C)CC)CC1C 21244,n1(CC)cc(CC(=O)N(C(C)CN(C(=O)Cc2cnc(C)s2)C)C)cn1 21245,C(N=c1ccnc(NCC2CCCCC2C)[nH]1)C1(OC)CC(C)(C)CC(C)(C)C1 21246,C(=O)(CC(C)(C)N(C(=O)CC1CCC=CCC1)C)N(CCCCCO)C 21247,c1(C(N(CCC(=O)NCCCNC(CC2C(C)C2)=O)C)=O)cnn2c1OCC2 21248,C1(C)(CNC(Cc2nc(CC)sc2)=O)CC(F)(F)CN1C(c1scnc1C)=O 21249,N1(C(C(CC)OC)=O)CCC(C)C(CNC(c2nccc(Cl)c2F)=O)C1 21250,c1(C2(C(=O)NC(CC=C)C3CC3)CCC2)ccc(F)cn1 21251,C1(NC(=O)CCOC2CCCC2)CC(O)(CNC(=O)CC2(C(F)F)CC2)C1 21252,C=CC1(NC(C23CC2CCN3C(c2sccc2F)=O)=O)CCCC1 21253,Cc1occc1CC(=O)NC1CCN(C(c2cn(C3CCCC3)nn2)=O)C1 21254,C#Cc1ccc(F)c(C(N2CCC(CNC(C3CCC(C)(C)OC3)=O)CC2)=O)c1 21255,c1(CC(N2CC=C(CNC(CC(C)F)=O)CC2)=O)ccc(S(N)(=O)=O)s1 21256,N1(C(C(C)Cc2ccccc2)=O)CC2CN(C(c3coc(O)n3)=O)CC2C1 21257,c1(C(N(C2CC(NC(c3ccc(Cl)cn3)=O)C2)C)=O)cnc2[nH]c(O)nc2c1 21258,c1(C(=O)NC(C(C)NC(C2CCCN2C=O)=O)CO)ccc(Cl)c(N)c1Cl 21259,c1(OC)ccc(CNC2CN(C(c3csc(C)c3C)=O)CC2C)c(C#N)c1 21260,C(CCN(C)C)(C(=O)NCc1cn(C)cn1)NC(COCCC)=O 21261,C=CC1CN(C(=O)C(C)(C)n2ccc(C)n2)CC1NC(=O)CC1C(=O)NN=C1C 21262,C(C)(CCCC(=O)N1CC(N2CCNC2=O)C1)NC(c1[nH]cc(C)c1C)=O 21263,C(=O)(C(CC(F)F)NC(c1ccc[n+]([O-])c1)=O)NC(CCC)CCO 21264,CCC(C)C(O)C(C)C(=O)NC1C2CCN(C(=O)C(O)C(C)(C)C)CC12 21265,C1(CNC(CCN(CCC)C)=O)C2CCCC1N(C(c1cccc(O)c1F)=O)C2 21266,C1(c2nnc(N(CC)CC3(O)CC(CS(C)(=O)=O)CC3)n2C)CC2(C1)CC(F)(F)C2 21267,CC1CN(C(C2(CC3CC3)CC2)=O)CCC1Nc1ccc(C#N)nc1 21268,c1(C(=O)NC23CCN(C(=O)CCn4ccnc4)CC2C3)ccc2[nH]ccc2c1F 21269,c1(C(N2CCCC(N(C(C(C)C3CCOC3)=O)C3CC3)C2)=O)ccc(Cl)nc1Cl 21270,C(c1ccc(C(F)(F)F)cc1)=CC(N1C(CNC(CCOCC#C)=O)CCC1)=O 21271,C#CCC(O)C(=O)NC(CCOCC)C(=O)NCCC1CCCCO1 21272,CC1(C)C(C)(NC(=O)C(F)CC2CN(C(=O)C(F)F)C2)C1(C)C 21273,CCC(CCOC)C(=O)NC1(Cc2cccc(C)n2)CC1 21274,Cc1c(NC(=O)CC2CCN(C(=O)Cc3cccnc3)CC2)cnn1C1CC1 21275,c1(C(N2CCC(COC)(NC(c3cncs3)=O)C2)=O)c(C)oc2nc(Cl)ccc12 21276,C(=O)(CC1=CCCC1)N1CCC(NC(c2c(C)oc(C(F)(F)F)n2)=O)C1C1CC1 21277,C1(C)(C(N2CC3(CC(NC(C4(OC)CC4)=O)C3)C2)=O)CCc2ccccc2C1 21278,C1(CNC(c2c(C)nc(CO)o2)=O)C2CCC(C2)N1C(=O)CCn1cccn1 21279,C1(C(=O)NCCC2CC(C)(C)C2)(NC(C(CCOC)C)=O)CCC(C)(C)C1 21280,C1(NC(CC(C)OC)=O)CCC(C)N(C(=O)C(CO)c2ccccc2)C1 21281,c1(C(=O)NC2CCN(C(CCc3ccc(C)cc3C)=O)C2)ccc2sncc2c1 21282,c1(C(=O)OC)ccc(Br)c(NNC(=O)C2Cc3c(F)cccc32)c1 21283,C(O)(CC(=O)NCC1(CC2CC2)CC1)(C(F)(F)F)c1ncc(C)o1 21284,c1(-n2cc(C(C)NC(C3CC3(Cl)Cl)=O)nn2)cccc(Br)c1 21285,C1(NC(C(CC)C)=O)CC(NC(c2sccc2CO)=O)C(O)C1 21286,N1(C(C2C(C)(C(F)F)C2)=O)CCCCCC(NC(=O)C2=CCCS2)C1 21287,CCCCC(C)CCC(=O)NCC1CC1CNC(=O)CC#N 21288,c1(C(C(=O)N(CC(C)NC(CNC(CCCCC)=O)=O)C)=O)cc(F)cc(Cl)c1 21289,Cc1nn(C)c(C)c1CC(=O)NC1CN(C(c2nccc(N)c2Cl)=O)CC1O 21290,N1(OCC)CCCCC1C(=O)NN(C(C1C(Cc2nnnn2C)C1)=O)C 21291,CC1CN2CCN1C(=O)C1(CCC1)C2=O.c1(NC(=O)C(C)(C)C)ccccc1F 21292,CC(C)(O)C(F)C(=O)N1CCOC(CNC(C2CCCCO2)=O)C1 21293,C(=O)(CCOCCCNC(=O)Cc1ccsn1)NCC(=O)N(C)CC 21294,c1(OC)cccc(-c2cc(C(=O)NCC=CCNC(c3sccc3CO)=O)on2)c1 21295,c1(C(=O)NC(C2CC2C(=O)N(CC(O)CO)CCO)C)csnc1Cl 21296,C1(NC(=O)NC(C2CCO2)C)CCC(F)(F)CC1(C)C 21297,S(=O)(=O)(c1cnn(C)c1)NCC(=O)N(CCCNC(=O)CC1COCCN1C)C 21298,C1(NC(COC2(C)CCCC2)=O)CC2C(NC(c3nocc3Cl)=O)C2C1 21299,CC1(C)OCc2c1n[nH]c2C(=O)NCC1CC(NC(=O)C(F)CC2CCCC2)C1 21300,c1(C(=O)NC2C(NC(COCCCCC)=O)CCC2)c2ccccc2nn1C 21301,c1(OCC(=O)N(C2CN(C(=O)CC(C)(C)N(C)C)C2)C)ccc(Cl)nc1 21302,CC(CNC(=O)C(F)n1cccn1)(CO)NC(C1(c2cccnc2)CC1)=O 21303,c1(C(N2CCCC(NC(C(C)S(N)(=O)=O)=O)C2C)=O)c(Cl)oc2ccccc12 21304,C(=O)(C1CCOc2ccccc21)NCC(C1CCCN1C(C1C=CCC1)=O)(C)C 21305,C(CC(=O)NC(C)CCCCO)(C(C)C)NC(C1(OCC)CCCC1)=O 21306,c1(C(=O)NC2(COC)CCN(C(C3(C)CCCN3C)=O)C2)ccnc(Cl)c1O 21307,C1(NC(C2(CNC(=O)CC3CCCC3)CCCO2)=O)CCCCCC1F 21308,c1(C(N2CC(C)OCC2C)=O)nc2ccccn2c1C1=CCOCC1 21309,c1(CNC(CSCC#C)=O)cc(C(=O)NCC2(C#N)CC2)no1 21310,c1(C(N2CCN(C(CC=C=C)=O)CC2C)=O)cc(Cl)cc2nc(C)[nH]c12 21311,N1(C(c2cnn(CC)n2)=O)CC(C2CCCCN(C(=O)CC3CC4(CC4)C3)C2)C1 21312,S(=O)(=O)(c1[nH]c(=NC2CCCC(C(C)(C)C)C2)ccc1Br)NCCCOC(C)C 21313,c1(C(=O)NCC2(CCNC(COC(C)C)=O)CC2)cncc2c(O)nccc12 21314,CCC(CC)CC(F)C(=O)NC(C12CCC(CC1)C2)CNC(=O)C(C)(C)O 21315,N1(C(CSCC)=O)CC2CCCCC2(NC(c2ccc(OC)cc2N)=O)C1 21316,C#CCC(O)C(=O)NCCCN(C(=O)C(O)(c1ccccc1)C1CCCCC1)C 21317,N1(C(C(CCC)CC)=O)CCCCCC(NC(=O)CN2CCC(C(N)=O)CC2)C1 21318,Cc1cncnc1N1CCC(C(C)(C)NC(=O)Cn2ccnn2)CC1 21319,C1(C(N(C(CC)C2CC2)C)=O)CC(F)CN1C(=O)CC1COCCO1 21320,C1(CNC(c2[nH]cc(CC)n2)=O)CC(C)CN(C(c2cncc(SC)c2)=O)C1 21321,NS(=O)(=O)C1(C(=O)NCC2(O)CCN(C(C3(n4cnnn4)CC3)=O)CC2)CCC1 21322,Cc1nc2ccc(C(=O)NCC3C4CN(C(c5csc(C)c5)=O)CC34)cc2s1 21323,N1(C(c2c(OC)ccs2)=O)CCC2(CC1)CC2NC(=O)C=CCOC1CCCC1 21324,O=S(=O)(c1ccc(NNC(=O)c2cccnc2)cc1)Nc1ccc(O)cc1 21325,C1(CCNC(c2cncc(CNC(C34C=CC(CC3)C4)=O)c2)=O)CCCCC1O 21326,C1(O)(CC=C)CCN(C(=O)C(CCCOC)NC(=O)C(C)NC(=O)NC)CC1 21327,c1(NC(N2CCC(CC(=O)OC)C2)=O)nc2ccccc2n1CC#N 21328,c1(C(=O)OCC)cc(CCNC(=O)Cc2nn[nH]n2)nc(O)c1 21329,CS(=O)(=O)c1ccnc(N(C(=O)CCN2CCCCC2)CC2(O)CCCNC2)n1 21330,C1(NC(CC2(C=C)CC2)=O)CC(=O)N(C2CN(C(=O)Cc3c[nH]ccc3=O)C2)C1 21331,C1(C)(C(=O)NC2(C(F)(F)F)CCCCO2)CCC(N(C)C(=O)OC(C)(C)C)C1 21332,C12CCOC1C(=O)N2.C1(NC(C(C)OCC)=O)CCCC1C(=O)OC 21333,C1(C(N2C(C(=O)NCC3CCOC3)CC=CC2)=O)CC2(C1)CC2(F)F 21334,C1(NC(=O)CCC2CC2)CCC2(CCN(C(c3csc(Cl)c3Cl)=O)CC2)C1 21335,c1(OC)cccc2scc(C(N3CC4CC(NC(=O)C(C)N(C)C)CC3C4)=O)c12 21336,N1(C(CCC#C)=O)CCC2CCC(C1)N2C(=O)CCOc1ccc(OCC)cc1 21337,C1(C2CCN(C(C3CCC(F)CC3)=O)CC2)(NC(C(CC)C(C)C)=O)CCC1 21338,C(CSc1nc(C)no1)(C(F)(F)F)NC(=O)OCC(=O)NCC.O 21339,c1(NC(C)=O)ccc(C(N2CCC(O)C(NC(=O)CCC(C)C)C2)=O)cc1Cl 21340,C12CC(N(C(=O)C3CC3)C1)C(=O)NCCN2.c1(COC)c[nH]c(C(=O)OC)c1 21341,C1(NC(C2(C)COC2)=O)CN(C(=O)C(C)(C)Cc2ccccc2)CCC1F 21342,CC(C(=O)NCC1CCN1C(c1cncc(C(F)(F)F)n1)=O)C(C)(F)F 21343,c1(C(N2C(CNC(=O)C(F)CC3CCC3)CCCC2)=O)cccc(C#CCO)c1 21344,C1(C(N2C3(CNC(C=CC(N)=O)=O)CCC3CC2)=O)CCC2(CC1)OCCO2 21345,C1(C)(C(N(CC(C)N(C)C(C2CCN(C)S2(=O)=O)=O)C)=O)CCC(F)(F)CC1 21346,C(=O)(CC(=O)NCCNC(c1cocc1C)=O)NCC 21347,N1(C(C2(NC(CC3C(C)CCC3)=O)CCOCC2)=O)CCN(C)CC(O)C1 21348,N1(C(C(C)(C)C(F)F)=O)CCCC(O)(CNC(C23CCC(C)(CO2)C3)=O)CC1 21349,c1(C(N2CCCCC2C(C)C)C(=O)NCCSC)cc2cccnc2s1 21350,c1(C(=O)NC2(CO)CN(C(C3CCS(=O)(=O)CC3)=O)C2)nccc2nn[nH]c12 21351,O=C(CCC(=O)C1CC1)NCC(O)CC(=O)NC1CCN(C2CC2)C1 21352,c1(C(N2CC(C)N(C(C3CCCC34CC4)=O)CC2)=O)cc2c(cn1)CCCC2 21353,c1(CNC(C2CCCN(C3CCC3)C2)C)ccc(I)c(F)c1 21354,C1(NC(C(CC)Oc2ccccc2)=O)CN(C(=O)CCC#N)CCC1(C)C 21355,C(=O)(CC(C)(C)CC(F)(F)F)N(N1CCCC(C2(N3CCNC3=O)CNC2)C1)C 21356,C1(NC(CCCc2cc(C)no2)=O)CCN(C(=O)C(C)SC(F)(F)F)CC1O 21357,C(=O)(C1CCCc2cncn21)NCC1C2CN(C(c3c(C)cc(N)cc3)=O)CC21 21358,c1(C(=O)NCC2CCN(C(C=C(C)C(F)F)=O)CC2)ccc2c(C)nn(C)c2n1 21359,c1(-c2cc(C(N3CCC(C)C3)=O)c(Cl)nc2)ccc(S(=O)(=O)NC2CC2)cc1 21360,C1(NC(c2n(C=C)ncc2)=O)CN(C(=O)C2=COCCO2)C(C)(COC)C1 21361,C1(C(N(C)CC2CCC(F)(F)C2)=O)CCCN(C(=O)Nc2ccc(Cl)cc2)C1 21362,Cn1[nH]c(=NC(=O)C2CCCN2C(C2(C(F)(F)F)CCC2)=O)cc1Cl 21363,C1(C(N2CC(C)C(F)C2)=O)N(C(c2cc(C(N)=O)c[nH]2)=O)CC12CCCC2 21364,N1(C(c2cc(COC)cn2C)=O)CCOC(C)(CNC(c2n[nH]c(C)c2Cl)=O)C1 21365,N1(C(Cc2c(C)n[nH]c2)=O)CC2CC(NC(c3nnn(C)c3N)=O)C(C2)C1 21366,N1(C(CS(CC)=O)=O)CC(S(=O)(=O)N2CCN(C(=O)C(C)(C)C#N)CC2)C1 21367,C(=O)(CCC(N)=O)NCc1c(C2CCN(C(C3(C)CC3)=O)C2)n[nH]c1 21368,C(c1cccc(C(F)(F)F)c1)=CC(=O)OCc1ccc(Br)nc1Cl 21369,C1(c2c(OC)cc(Br)c(F)c2)NC(=O)N(CCC2CC2)C2=C1C(=O)NC(C)C2 21370,C(=O)(CCc1ncc[nH]1)NCC1(NC(CN(C(C)=O)C)=O)CC1 21371,C1(CC=C)CCCN(C(=O)NCCNC(C2CCCCC2)=O)C1 21372,C1(NC(CCC2CCN(C(c3c(C)nc(C)o3)=O)C2)=O)CC2(CCCC2)C1 21373,C1(CCN(C)C(C2(C(F)F)CCCC2)=O)CCCCN1C(=O)CC1C=CCC1 21374,c1(C(=O)OCC(c2ccccc2)OCC)cc(N(C)C)oc1C 21375,N1(C(C2CN(C(c3ccc(N4CCC4)cc3)=O)CCS2)=O)CCc2nc[nH]c2C1 21376,c1(C(=O)NC(C)CCNC(=O)C=CC2CCCC2)cnc2ncnn2c1O 21377,N1(C(CSCCC#N)=O)CCN(C(C2CCC3(CC2)CC3)=O)CC1CC(F)F 21378,CCC(C(=O)N1CC(OCC(N)=O)C1)NC(c1cc(CO)[nH]n1)=O 21379,C1(NC(CC(CCC)C)=O)CCC2CN(C(=O)C(C)(C)C)CCC2C1 21380,n1(CC(=O)N(C)CC2CC2CF)nnnc1C1CC1.C12CN(C1)C2=O 21381,CC(C)(C)C(C#N)C(=O)NCCC1(C)CCN(C(C2CC3(CCC3)C2)=O)C1 21382,c1(CN(C(=O)NC2CC(CC(C)(C)C)C2)CC)cnn(CC)c1 21383,N1(C(C(C)OC)=O)CCC2CN(C(=O)CN3CCP(C)(=O)CC3)C2C1 21384,CCC(C)(C)CC(=O)NC1CCCC(NC(=O)CSCc2ccc(F)cc2)CC1 21385,N1(C(CCc2cc(C)no2)=O)CC(N(C(=O)C(F)OC(F)(F)F)C)C(O)C1 21386,C1(C(N2CC(OCC)(CNC(=O)C(C)C(C)CC)C2)=O)CC2CCC1CC2 21387,Cn1nc(C2CC2)cc1NC1(C(C)(F)F)CC1 21388,c1(OC)cccc(F)c1C1CCCN1CC(=O)Nc1ccnc(Cl)n1 21389,CC(C)CCCCC(=O)N1CC(C(=O)NCC2CC23CC3)CCC1(C)C 21390,Cc1cc(C(C)NC(=O)N(C2CC=CCC2)CCO)no1 21391,CN1CCN(C)C(C(N2CCOCC2C(=O)NC2CCCC2O)=O)C1 21392,n1(CC2(C(=O)NCC3CC(CNC(C(C)N(C)C)=O)C3)CC2)cc(C2CCC2)nn1 21393,C=C=CC(C)C(=O)NC1(C)CCN(C(C2CC(=C3CCC3)C2)=O)C1 21394,Cc1csc2ccc(C(N3CCCC3(C)CNC(=O)C(C)N(C)C)=O)cc12 21395,N1(C(CCC(CC)C)=O)CC2(CCC(NC(=O)C(O)CSC)CC2)C1 21396,C12(CNC(CC3OCC(C)(C)OC3)=O)CCC(CC1)N(C(=O)C=C1CCC1)C2 21397,C(=O)(NNc1ccc(C(=O)O)cn1)c1c(CC)[nH]cc1 21398,c1(N2CCC(C)(CC)C2)ccc(S(=O)(=O)NCC(c2ncccc2F)(C)C)cn1 21399,CCC(C)(C)C(O)C(=O)N1CCC(CCNC(=O)C(c2ccc(F)c(F)c2)O)C1 21400,c1(CC(=O)NCCNC(c2cc(F)cc(N)c2F)=O)ccc(S(=O)C2CC2)cc1 21401,Cc1ccc(C)c(C(N2CC(CNC(=O)CC=CC(C)(C)C)C(O)C2)=O)c1 21402,C1(NC(CC2(C)N(C(c3ccc(C)s3)=O)CCC2)=O)CC2CC3C(C2)C13 21403,c1(CCC)cc(C(=O)NC2CC(CNC(C3(C)C=CCCC3)=O)C2)ccn1 21404,C1(C(=O)OC)CCN(C(=O)C(C)NC(c2c[nH]nc2C(C)C)=O)CC1 21405,c1(CNC(NC(COC)C(C)C=C(C)C)=NCCCF)cc2c(cc1Cl)OCCO2 21406,C1(NC(CCC=CC)=O)CCCN(C(c2cn(C3COC3)nn2)=O)C1C 21407,CN1CCCC(C(N2CCCC(n3cc(COCCO)nn3)C2)=O)C1 21408,c1(CC(=O)NCC2CC(NC(c3ccsn3)=O)C2)ccc(OC(F)F)cc1 21409,C1(C(=O)NC(C(C)CN(C2CCCC2)C(CNC(CC)=O)=O)(C)C)CCCN1N=O 21410,C1(OC(N(C)C)=O)C2CCN(C(=O)C(=O)N)C2C1(C)C.c1(C)n[nH]c2c1CCCC2 21411,c1(C(N2C(C)(C(=O)Nc3ncnc(Cl)c3C(N)=O)CC2)=O)ccc(F)cc1C#N 21412,C(CCC(C)(C)C(=O)NC(c1nccn1C)CC)NC(C(CCCC)O)=O 21413,C1(CNC(=O)CCOC2CCOC2)CCCN(C(c2cc[nH]c2)=O)CC1 21414,c1(NC(c2ccc(-n3ncc(C)c3)cc2)=O)ccc(Cl)c(Br)c1Cl 21415,N1(C(CSCC#C)=O)C2CCC1CN(C(=O)C(C)SCc1ccccn1)C2 21416,C1(C(=O)NC(C)CN2CCN(C(C3CC4(CSC4)C3)=O)CC2)CCC(=O)C(C)C1 21417,N#CC1CCN(C(=O)CC2(NC(=O)CC3CCOC3)CC2)C1 21418,c1(C(N2CCC(NC(CCCN(C)C)=O)(CO)CC2)=O)ccc2nonc2c1 21419,CC1CC(NC(c2ccoc2Cl)=O)CN1C(c1c[nH]c(C(F)(F)F)c1)=O 21420,O(N1C(=O)c2ccccc2C1=O)CC(=O)NC(C)CNC(C1(F)CCCCC1)=O 21421,c1(CC)nc(CC(=O)N(C)CCN(C)C(C2CC2(C)C)=O)cs1 21422,N1(C(C2N(N=O)CCC2)=O)CC(NC(=O)C(F)(F)C(F)(F)F)CC2(CC2)C1 21423,N1(C(C(C)(C)NCC)=O)CCC(C=CC(=O)NOC(C)C)CC1 21424,c1(OC)cc(C(=O)NC2CN(C(=O)CC3CC3C3CC3)CC2F)c(Cl)cc1Cl 21425,C1(NC(C=C(CC)C)=O)CC2(C1)CC(NC(C1CCC(C)(CC)O1)=O)C2 21426,C1(NC(Cc2cccc(OC)c2)=O)CCCN(C(=O)CS(C)(=O)=O)CC1 21427,N1(C(C(=O)N(CCOCC2CC2)C2CC2)CC2CCCC2)CCCC(F)CC1 21428,C(=O)(C(C)(F)C(C)(C)F)NC(CCC)C(=O)Nc1ccc(F)c(C(=O)O)c1 21429,CC1=CC(NC(=O)CCC2CC(NC(=O)Cc3ccns3)C2)CCC1 21430,N1(C(CC(CC)O)=O)CCOCC(CNC(c2ccc(C3CC3)nc2O)=O)C1 21431,C1(N(C(C2(CC=C)CC=CC2)=O)C)CCCN(C(=O)Cc2nccc(OC)n2)C1 21432,CC(CCNC(C1(S(C)(=O)=O)CC1)=O)CCNC(=O)CSC1CC1 21433,c1(C(N2CCC3CN(C(C(CC=C)CC=C)=O)CC32)=O)cccc2oc(O)nc12 21434,c1(OC)cc(OC)cc(C(N2CC3(NC(=O)CC4CSC4)CC2C3)=O)c1 21435,C(C(CO)C(C)(C)C)NC(C(C1CCCC1)NC(c1nn(C)c(O)c1)=O)=O 21436,c1(N2CCC(=C)C2)ccc(S(=O)(=O)NCCN2CC3CC3C2)cc1Cl 21437,c1(C(c2n(CCC)nnn2)NCC(c2ccccc2F)C)noc2c1CCC2 21438,N1(C(CCCCC=CC)=O)CC(NC(=O)C(=C2CCCCC2)F)CC(C)(C)C1 21439,c1(C(=O)NCC(C)N(C(c2cnc(O)n2C)=O)CC)c(C)cncc1C 21440,N1(C(c2c(C)cn(C)c2)=O)Cc2[nH]nc(C(N3CC(O)(C(N)=O)C3)=O)c2C1 21441,C(=O)(CCCC(=O)NOC(C)(C)C)NCC(CC)NC(CC=C(C)C)=O 21442,C1(NC(c2cnnn2C2CC2)=O)CC2CC(C1)N(C(C1SC3C=CC1CC3)=O)C2 21443,c1(C(N(CC2N(C(c3cn(CCC=C)nn3)=O)CCC2)CC)=O)cc(Cl)cn1C 21444,N1(CCCC(C)(F)F)CCC2C(O)CC2C1 21445,N1(C(c2cn(CC=C)nn2)=O)CCCC2(CC(NC(C3CC(F)(CO)C3)=O)C2)C1 21446,C(C(F)(C(=O)N1CCCCC1C(C)C)C(C)C)NC(c1nc(CC)oc1)=O 21447,N1(c2cc(NCc3c(COC)noc3)nc(C)n2)CCC(CC#N)C(F)(F)CC1 21448,N1(C(C2(C)COC2)=O)CC2(CCCCN2C(=O)CN2CCNC2=O)C1 21449,c1(OC)cnccc1C(=O)NC1CCCCC1NC(=O)COCCSC 21450,C1(NC(CCC2(C(=O)OC)CCCC2)=O)CN(C(C2CCOC2C)=O)CC1C 21451,C12(C(=O)NC3CCC(CNC(c4c[nH]nc4F)=O)CC3)CCC(CF)(CC1)CC2 21452,N1(C(c2ccn(COC)n2)=O)CCN(C(=O)CNC(c2cc(CF)on2)=O)CC1 21453,c1(CCC(=O)N(C2CN(C(C3CNC(=O)C3)=O)C2)C)nc(-c2ccco2)no1 21454,C=CCC(CNC(=O)CC(CC)C1CCC1)C(=O)NC(c1ncc[nH]1)C 21455,c1(C(=O)NC(CC)CNC(=O)CC(C)C2CCCCC2)nccc2cccnc12 21456,C1(NC(c2c(OC(C)C)nccc2)=O)CN(C(C2CCC3CC23)=O)CC2(CC2)C1 21457,C1(NC(COCC(C)(C)C)=O)CN(C(=O)Cc2ccsc2)CC2CC12 21458,O(NC(=O)C(CC#CC)NC(=O)C=Cc1ccncc1)Cc1ccc(C#C)cc1 21459,c1(C(=O)NCC(CC)NC(c2cccc(N)c2C)=O)cccc2[nH]cc(Cl)c12 21460,c1(C(N2CCCC(CC(=O)NC3CCC(C)CC3)C2)=O)c(F)cc(O)cc1F 21461,c1(C(C)C)noc(CCC(=O)N2CCC2CNC(=O)C(F)(F)c2nccs2)n1 21462,c1(C(=O)NC2C(C)N(C(=O)C(C)S(C)(=O)=O)CCC2)cnc2cc[nH]c2c1 21463,N1(C(C(=Cc2cnc[nH]2)C)=O)CCN(C)C(CNC(=O)C(C2CCC(=O)N2)C)C1 21464,Cc1cc(CN(C(=O)C(C2(C)CC2)NC(c2nccn2C)=O)C)n(C)n1 21465,C(=O)(C(CCOC)NC(C1CCN(C)C1C)=O)N1CC(N(CC)CC)C1 21466,c1(C(=O)NC(C2CCN(C(c3cc(C)sn3)=O)C2)C)cccc(=O)n1O 21467,c1(C(C)NC(=O)NCC(=O)NCC2CCOC2)ccncc1F 21468,C(=O)(C1CCCc2cncn21)NC(C)CCNC(=O)C(c1cc(F)cc(F)c1)O 21469,C1(NC(CN(C(=O)CSC)CCOC)=O)CC(N(C)C)C(O)C1 21470,c1(CCC(=O)N(C)Cc2ccccc2Br)cccc(OC(F)(F)C(F)F)c1 21471,C1(COC(C)C(=O)NC2(CCNC(c3cc(C(F)F)cs3)=O)CC2)CCCCO1 21472,C(=O)(C1=CC(O)C(NC(=O)CN2CC3CCC2C3)C1)NC(CCC(C)C)C 21473,C(C)(C)(CCC(=O)N1CCC(c2ccccc2)(C(=O)NCC2CC2Cl)CC1)OC 21474,C1(C(=O)NCC(CNC(=O)CC(F)(F)Cl)F)COc2ccccc2C1 21475,C1(O)(C(C)NC(c2csc(Cl)n2)=O)CCN(C(C2CCN(C)C2=O)=O)CC1 21476,N=c1cc(C(N2CCNCC2CF)=O)c2ccccc2[nH]1 21477,C1(C)(CNC(CC)=O)CN(C(C23CCCC2CCC3)=O)CC1C 21478,c1(CN2C(C(N3CC4CCC(C3)O4)=O)CC(OC)C2)cccc2[nH]nc(O)c12 21479,N(C1CCCc2n[nH]cc21)C(c1c(C(=O)OC)c(F)ccc1Br)=O 21480,c1(N(C)CC2CCCC(O)C2)cccc2c(Br)cncc12 21481,C1(NC(C(C)c2ccsn2)=O)CN(C(c2ccnnc2O)=O)C(C)(C)C1 21482,c1(C(=O)NC2CCN(C(C(C(C)C)NC=O)=O)C2)cccc2nc(O)oc12 21483,C1(CCCNC(C=CC=CCC)=O)CCCN1C(c1cc(C)c[nH]1)=O 21484,C1(COC2CN(C(=O)NC(C)C(N3CCC(O)CC3)=O)C2)CC(C)(C)OC1(C)C 21485,C(=O)(C#CC1(C)CCCO1)NCC1CCN(C(C(C=C=C)C)=O)CC1CC 21486,C1(NC(CN2CCC(C)CC2)=O)CC2CC1CC2C(=O)NCCCc1cccs1 21487,C1(C)(C(=O)NC(C=C)C2CC2)CCN(C(=O)COC2(C)CCC2)C1 21488,N1(C(CS(=O)(=O)NCC)=O)CCN(C(c2scc(C)c2C)=O)CC1CC 21489,Cc1cc(Cl)ccc1NC(C1CSCN1C(=O)C(C)c1cc[nH]n1)=O 21490,N1(C(CN(C2(CC)CCCC2)C(=O)OCC)=O)CC(CC)(CC)C1 21491,c1(CN2CCC(C)(NC(C3CN(CCC)C(=O)C3)=O)C2)n[nH]c2ccccc12 21492,c1(C(NN2C(C)Cc3ccccc32)=O)cccc(S(=O)(=O)N=S(C)(C)=O)c1 21493,C1(C(=O)NC2(C)CCCCC2)CCC2(CCN(C(C3CCNC(=O)C3)=O)CC2)O1 21494,N1(C(CCSCC)=O)CCC2CN(C(=O)CC34CCCC3C4)CC2CC1 21495,c1(C(=O)NC2(CF)CCN(C(C3CC(C#N)(O)C3)=O)C2)ccnc2[nH]nnc12 21496,CC1(C)NC(=O)CC1C(=O)NC12CC(C1)N(C(=O)Cn1cc(C3CC3)nn1)C2 21497,c1(OC)ccc2c(c1)OCC(CN1CCCC(CCO)CC1)=C2 21498,C12(C(=O)NCC(CNC(c3[nH]cc(C(=O)OC)c3)=O)(C)C)COC(CCO1)C2 21499,C1(C(=O)NCC(CC(=O)NC)C)CCN(C(c2occc2C(C)C)=O)CCO1 21500,C(=O)(C#CC1(C)CCCO1)NCC(C)CNC(c1ccccc1C1CC1)=O 21501,C1(F)(C(=O)NC2CC(CCNC(C=CC(C)C)=O)C2)CCCOC1 21502,N1(c2c(C(=O)OC)cc(C)cn2)CCC2(CCCCC2NC(=O)CC2CC2)C1 21503,CCC1=C(C(=O)N2CCN(C(c3c(C)cnn3C(C)C)=O)C(COC)C2)SCCO1 21504,C=CCC(CC(C)C)C(=O)N1CCN(C(=O)Cc2ncoc2C)CC12CCC2 21505,c1(CC(=O)NC(C)CC(C)NC(c2ncoc2C2CC2)=O)ccc(F)c(Cl)c1F 21506,N1(C(C(CNC(C2(C)CC(=C)C2)=O)C)=O)CC(C)C(C)C1C 21507,C(C(C)(C)CCNC(=O)C(C1CCCN(C(c2cnc(=N)[nH]c2)=O)C1)C)OC 21508,c1(C(=O)NC(c2cccnc2)C(N2CCC(CO)C(O)C2)=O)cnn2ccccc12 21509,N1(C(CCSc2nnc(C(=O)NCCN(CC)CC)o2)=O)CCNC(=O)C1 21510,Brc1c[nH]c2c(-c3nc(CC4CC4)nn3Cc3ccncc3)cnn12 21511,C1(CNC(C(CC)(C)COC)=O)CCC2(CN(C(c3cc(F)cc(Cl)c3)=O)C2)O1 21512,C1(NC(C2CC(C)(C)OC2)=O)CCN(c2ccc(C#N)nn2)CC1O 21513,C1(C(N(C2CCCN(C(=O)CC3COCC(C)(C)O3)C2)C)=O)CC(=O)CC(=O)N1 21514,C1(NC(C(=Cc2cccnc2)C)=O)C2CCC1CN(C(c1ccns1)=O)C2 21515,O=C(C(Cc1ccoc1)NC(C1CC1(F)F)=O)NCC(F)(F)CC1CC1 21516,Cn1ncc(Cl)c1-c1cc(C(N2CC(c3cn(CC4COC(=O)C4)nn3)C2)=O)on1 21517,C(=O)(C1CCCc2nn[nH]c21)NCC(CNC(=O)COC1CCCOC1)O 21518,C1(C(=O)NCc2ccc(C(=O)OCC)o2)C(Cl)(Cl)C12CC2 21519,C1(C2CC2)(NC(C(c2cccc(C)c2)C)=O)CCN(C(=O)CCN(C)CCO)C1 21520,N1(C(CC2CCN(C(CC3C(CC)C3)=O)C2)=O)CCC(C2CCC2)C1 21521,c1(C(=O)NC2(CC=C)CCN(C(=O)CC3(O)CCCC3)C2)cc(OC)nc(F)c1 21522,Cc1cccc2c1CCCN2C(=O)NCC1COC(C)(C)OC1 21523,c1(CC(=O)N(C(C(=O)N(CC(O)CF)CC)C)CC)ccc(C)nc1 21524,c1(C(=O)OC)ccc(CN2CC3C(CNC(=O)CC(=O)OC)C3C2)cn1 21525,C1(CC(=O)NCCC2CN(C(C(C)Oc3ccccc3)=O)C2)CC2CCC1CC2 21526,c1(C(=O)NC(CCNC(C(C(CC)C)O)=O)C)c[nH]c2cccnc2c1=O 21527,N1(C(CC(=O)N(C)C)=O)CCCC2C(NC(=O)Cc3cn[nH]c3)C(C)(C)C12 21528,N#Cc1ccc2c(c1)C(=Cc1cnc(CO)cn1)CC2 21529,C=CCC(O)(CC=C)C(C)NC(C1(C)CNC(=O)N1)=O 21530,C(=O)(C1=NOCC1)N1CC(C(=O)NOC(C)CC)(CC=C)C1 21531,C(=O)(CCCCCN1CCOCC1)NC(c1cn(CCO)nn1)CCC 21532,C1(C(CNC(C23CCC2C3)=O)F)CCN(C(=O)C(F)(F)C2CC2)CC1 21533,N1(C(C2(OC)CC2)=O)CC=CC(NC(c2c[nH]nc2C2CC2)=O)C1 21534,CC(C)C(CNC(C1CC2CCCC2C1)=O)C(=O)NCC(C)(F)C(C)(C)F 21535,C1(O)(CNC(C(CNC(C=C=C(C)C)=O)OC)=O)CC2C=CC1C2 21536,c1(C(=O)NC23CC2CN(C(c2csc(CC(F)(F)F)n2)=O)C3)coc2c1COC2 21537,C1(C)(C(=O)NC(C2CCCO2)CC)CN(C(=O)CCCCNC(C)=O)C(C)(C)C1 21538,N1(C(C(CC)F)=O)CCN(C(C2(C)CCC(=O)C2)=O)CCC1C 21539,C=CCCC(F)(F)C(=O)NC(CO)CCCCNC(c1cnsn1)=O 21540,c1(C(C(=O)N(CCN(C(CC2(C=C)CC2)=O)C(C)C)C)(C)OC)ccccc1F 21541,CCCCCCC(C)C(=O)NC1CC1NC(c1cc(C)cc(F)c1N)=O 21542,c1(C(=O)NC(CNC(Cc2c(C)non2)=O)CO)ncc[nH]c1=O 21543,c1(-c2cn(CC(N3CCCC3CN3CCCC3)=O)nn2)cccc(OC(F)F)n1 21544,C1(CNC(CC(CC)OC)=O)CN(C(=O)CCc2nc(C)no2)CCC1(F)F 21545,N1(C(c2ccc(CN(CC)CC)o2)=O)CC(CCNC(c2ccsc2)=O)C(C)C1 21546,c1(C(=O)Nc2c(C)ncc([N+](=O)[O-])c2)ccc2ncc(Br)cc2c1 21547,c1(C(=O)NC(CNC(C2CCC3CC23)=O)CO)cc2c(c([N+](=O)[O-])c1)OCO2 21548,n1(CC)nc(C)c2cc(C(=O)NCC(C)(CO)NC(C3CC4CCC4C3)=O)sc12 21549,N1(CC)CC(NCc2cnc(Cl)c(F)c2)CC(C)C1 21550,N#Cc1ccnc(N2CCCC(C(N3C4CCC3C(N)C4)=O)CC2)c1 21551,C1(COC)CN(C(=O)C=Cc2cccs2)CCN1C(=O)CC(C)(C)F 21552,C=CCC(C)(C)CC(=O)NC(CNC(c1ccc(OCCN(C)C)cc1)=O)CO 21553,C1(CCNC(C2C(C(=O)OC)CCC2)=O)CCN(C(c2nc(O)c(C)s2)=O)CC1 21554,C1(C2CCN(C(=O)CCCCC(F)F)C2)(NC(=O)Cn2cc(CO)nn2)CC1 21555,N1(C(COCCCOC)=O)CCC2(CC1)CCN(C(C1CCCC1OC)=O)C2 21556,c1(CC(C(=O)NCC(CNC(Cc2nc(C)[nH]n2)=O)CO)C)ccccc1F 21557,c1(C(=O)NC2C(C)(C)N(C(C3CN4CCN3CC4)=O)CC2)cnc2nccn2c1 21558,CC1C(C)N(C(=O)C2=CCCOCC2)CCN1C(=O)C(O)CC1CCCC1 21559,c1(CC(=O)NCC2(O)CN(C(c3oc(C)c(CO)c3)=O)C2)cccc([N+](=O)[O-])c1 21560,CC(C)C(C(=O)NCC(n1cc(-c2cccc(C(F)(F)F)c2)nn1)C)C(C)C 21561,S(=O)(=O)(c1ccc(Cl)nc1C)N1CC2(CN(C(C(CC)O)=O)C2)C1 21562,N1(C(CCOC2CN(C(c3snc(C)c3N)=O)C2)=O)CC2CC(C)(C)C2C1 21563,C(C(CC(C)C)C(=O)NCc1c(C)noc1C)NC(C=CCN(CC)CC)=O 21564,c1(OC)ccc(C(=O)NCC(CNC(=O)CCc2cccnc2F)CO)c(C)c1 21565,CC1(C)COCCC1CNC(C1CCCN1Cc1sccc1Cl)=O 21566,c1(SCC(=O)NC2CCCC2NC(c2csc(CO)n2)=O)ccc(F)cc1F 21567,C1(CC=C)(NC(=O)CCc2ccc(C)s2)CCN(C(C2CCO2)=O)C1 21568,c1(C(N2C(CN(C)C(c3ccon3)=O)COCC2)=O)noc2c1CCCCC2 21569,C1(C(=O)NCCOC2CN(C(C(C)(C)C)=O)C2)Cc2ccccc2O1 21570,Cc1scnc1C(=O)NCC(C)C(=O)NCCN1CC2CC2C1 21571,C=C(Br)CC(=O)NC(C1(O)CN(C(c2ncn(C)n2)=O)C1)C 21572,N1(C(=O)Cc2cncc(F)c2)CC2CC(C1)N(C(=O)COc1cccnc1)C2 21573,OC1(CNC2CCN(Cc3ccccc3)C2)CC(O)C1 21574,Cc1cc(C(=O)NC2CN(C(c3cnco3)=O)CCC2C)c2cccnc2c1C 21575,CCC(CC(=O)NCCCOCCC(=O)NC1C(CO)CC1O)C(C)C 21576,CC1=CC(NC(=O)COC(C)(C)CNC(C2(C)CCCC2)=O)CCC1 21577,CN1CCN(C(C2COCC2NC(=O)C=Cc2cocn2)=O)CC1=O 21578,c1(C(N2CCN(C(C3(C(=O)NC)CCC3)=O)CC2)=O)cncc(Br)c1C 21579,N1(C(c2cscc2C)C(=O)NC2(C(=O)OC)CCCC2)CCn2ncc(Cl)c2C1 21580,C(CCC(=O)NCC1CC1NC(=O)Cc1ncoc1C)=C(C)C 21581,Cc1[nH]c(C)c(C(=O)N(N2CCC(c3ccccc3)(C(F)(F)F)C2)C)c1C 21582,CN1CCc2ccc(NC(=O)Nc3ccc(-c4nncn4C)cc3)cc21 21583,C1(C(N2CC(C3CCOCC3)C2)=O)CCOCC1C(N1CC=CC1)=O 21584,CC1(C(=O)NC2CC(CNC(=O)CC3CCCC34CC4)C2)CC(C#N)C1 21585,CC1CN(C(c2cnc(CNC(=O)C3=CCCCO3)nc2)=O)CC(C)(C)O1 21586,c1(OCC)nn(C)cc1C(N1CCC(N(c2cc(C(C)C)ncn2)C)CC1)=O 21587,C(CCC(CO)NC(=O)CC1CC(O)C1(C)C)NC(c1nc(COC)oc1)=O 21588,N1(C(Cn2c3cccc(C)c3cc2)=O)CCC2(NC(=O)CCF)CCCCCC12 21589,C(=O)(C1=CCCSC1)N(CCCSc1cccs1)C(=O)CC1CCNC1.CO 21590,C1(C(N(C2CCCC2)CC(C)C)=O)COCC1NC(=O)CCc1cnn(C)c1 21591,c1(C(C)OC(=O)COC(=O)Cc2cn(Cc3cc(C(F)F)no3)nn2)nnnn1C 21592,Nc1cc(C(N2CC(NC(=O)CCNC(c3ccsc3)=O)C2)=O)cc(F)c1 21593,CC(C(=O)NCCN(C)C(c1ccns1)=O)C(F)F 21594,c1(-c2ccc(C(=O)NC(CNC(C=C(CCC)C)=O)C(C)C)[nH]2)ccc(Cl)cc1 21595,N1(C(C(Cn2ccc(C)n2)C)=O)CC2CCN(C(c3n[nH]cc3C)=O)CC2C1 21596,Cc1cc(Cl)ncc1NC(=O)CC(O)CNC(=O)CC1CCCN(C)C1 21597,c1(C(N2CCC(NC(CCS(C)=O)=O)(CO)CC2)=O)ccc2c(c1)CC(=O)N2 21598,C1(COC)CCC(N(C(=O)C(C)N(C(=O)C=C2CCOCC2)C2CC2)C)C1 21599,CCC1=C(C(=O)NC2CC(NC(c3cc(NC(C)=O)cnc3C)=O)C2)CCCO1 21600,N1(C(CN(C(=O)OC)C)=O)CCCC(NC(=O)CCc2cscn2)CC1 21601,CC1C2CCC(C2)C1C(N1CCCC(C)(C(=O)NC2CC23CCOCC3)C1)=O 21602,C1(CCNC(C(C)NC(CC)=O)=O)CCN(C(c2cn(C)cn2)=O)C1 21603,C(C(CC(F)(F)F)NC(C1(C)CC1(Cl)Cl)=O)NC(c1c(CC)oc(C)c1)=O 21604,O(NC(=O)CCC1(CNC(=O)CC2CCNC2=O)CC1)CC(=O)OCC 21605,Cn1ncc2cc(C(N3CC(NC(=O)CC4CCCOC4)C(F)C3)=O)cnc12 21606,N1(C(c2cc(CC)ncc2)=O)CCC2CCCC12C(=O)NC1CCCC(C)(C)C1 21607,C1(CNC(CCC)=O)CCN(C(C2CCC3CC2CO3)=O)CCC1(F)F 21608,N1(C(c2ccc(C)c(Cl)c2)=O)CCOCC12COCCN(C(=O)C1=CCC1)C2 21609,c1(C(=O)NC(CNC(c2cc(C)no2)=O)CO)ccn2ncc(Br)c2c1 21610,c1(C(N2CCC(CN(C(C(C=C)O)=O)C)CC2)=O)ccc(S(=O)(=O)CC)cc1N 21611,C(C(=O)NCC1CC2(CCC2)CN1C(=O)CC(C)CF)(c1ccccc1)=C(C)C 21612,N1(C(C(C)NC2(CO)CCCC2)=O)CCC(N(C(=O)C(C)(O)C2CC2)C)CC1 21613,C(=O)(C(C)(C)CCCC(C)=O)NC(CCCC)CCC 21614,c1(C(N2CCN(C(C(COC)C)=O)CC2CO)=O)ccc2c(c1)CC(C)(C)C2 21615,c1(CNC(N2CCCN(CCN(C)C)CC2)=O)cccc2cccn12 21616,c1(N2CCCC(N(C(=O)C(C)(C)C(F)(F)F)C)CC2)nc2ccc(F)cc2s1 21617,c1(-c2nc(CCOC)nn2-c2ccn(C(C)C)n2)c[nH]c2cccnc2c1=O 21618,C1(C(=O)NC2C3CCN(C(=O)Cn4cccn4)C23)C2C3CC4C1C1C2CC3C41 21619,Cc1cc(Nc2ccc(-c3noc(-c4c[nH]cc4Br)n3)nc2)ccc1F 21620,N1(C(c2cc(C)c(C)s2)=O)CCC2(CC1)CC2NC(c1nnc(C)cc1O)=O 21621,N1(C(C2OCC3CCCC23)=O)CC(O)CC2(CCOCC2)C1 21622,c1(C(=O)NC2CN(C(c3cocn3)=O)C3CC23)ccc(-n2cccn2)cc1Cl 21623,N1(C(CCn2ccc(C)n2)=O)CCCCC(CNC(=O)CC2COCCN2C)C1 21624,c1(CCC(=O)OC(c2noc(N(C)C)n2)C)csc2nc(C3CC3)cn12 21625,c1(CC)c[nH]nc1C(=O)N(CC(C)N(C(=O)CCc1cccnc1)C)C 21626,C1(CNC(C2C(C=C)C2)=O)CN(C(=O)CCC(=O)OCC)CC12CC2 21627,C1(C)(C(N2CCC(N(C(=O)C=CCOCCOC)CC)C2)=O)CNC(=O)C1 21628,N(C1CCc2cc(Cl)ccc21)c1ccc(NC(C)=O)c(C(F)(F)F)c1 21629,N1(C(C(CC)CCOC)=O)CCC2(CC2)CC1C(=O)NCC(C)(O)CO 21630,CC(C)CCN(C(=O)C(C1(O)CCC1)CCNC(=O)OC(C)(C)C)CC(C)C 21631,c1(OC)ncccc1C(=O)N(CC(C)NC(c1ccc(-c2ccccn2)o1)=O)C 21632,c1(OC)cc(Cl)c(CNC(c2nccn2Cc2cccnc2)=O)cc1Cl 21633,C1(C)(C(N(CC(C)CNC(=O)CN2CC(C)(C)C2)C)=O)CCC(=O)N(C)C1 21634,C1(COC)(NC(C2CC3CC3C2)=O)CCN(C(c2ccnc(C)c2)=O)CC1 21635,NCC(Cc1ccc(F)cc1)C(=O)N1CCC(CC#N)CC1 21636,c1(C(=O)NCC(C2CCCOC2)OCC)cnc2ccccn12 21637,C1(CNC(CCC(=O)NC)=O)CN(C(=O)CC(C)(F)F)CC12CCC2 21638,C1(C(=O)NCCc2scc(C(C)C)n2)CCCC1S(C)(=O)=O 21639,c1(C(N2CCCC2c2ccc(Cl)s2)=O)cc(CCc2cn(CC3CC3)nn2)on1 21640,C=Cc1cc(C(=O)NC(CO)C(C)NC(c2csc3nccn23)=O)cc(F)c1 21641,n1(C2CCC(C)C2)nc(CC2CCCC2)nc1C12CC(C1)C2 21642,C(c1ccccc1F)=CC(=O)NC1CC(CCNC(C2CC3(C2)CC3F)=O)C1 21643,c1(C(C(=O)N(CCOCC)NC)N(C2CCC(C(F)(F)F)CC2)C)sc(C)nc1C 21644,C1(C(=O)NCCCCCOC)CCN(C(=O)C2=C(C)CC2)C1C(C)C 21645,CC1(C(N2CCCC(CNC(=O)COc3ccccc3F)C2)=O)CCC(F)(F)C1 21646,C12CCCCN1C(=O)C2.CC1(NC(=O)CSC)CN(C(C2CCCS2(=O)=O)=O)C1 21647,N1(C(CSCCOC)=O)CCOC(c2cn(CCCC3CCOC3)nn2)C1 21648,c1(-c2nc(C3CCCC(=O)O3)n(C3CCCSC3)n2)cc(F)cc(F)c1 21649,N1(C(c2ccn(CC#N)n2)=O)CCC(CNC(c2cccc(C(F)F)c2)=O)CC1 21650,c1(C(N2C(CC)CN(C(c3cc(Br)cn3C)=O)CC2)=O)ccc2n[nH]cc2c1 21651,C1(CCCCNC(C(C=CC)O)=O)CCN(C(=O)CCSC)CC1 21652,C1(C(=O)NC(c2cccs2)C)C=CCN1C(C1(C)CCCO1)=O 21653,CC1=NNC(=O)C1CC(=O)NCC1(CNC(C2(C)CCOCC2)=O)CC1 21654,C(=O)(C(F)(F)CCn1cccn1)NCC(C)CN(C)C(c1cc(=O)cc[nH]1)=O 21655,c1(C(N2CC(CCNC(C=CC(C)C)=O)OCC2)=O)cccc2c1C(C#N)C2 21656,N1(C(C2C(CC(C)C)C2)=O)CCC(O)(CCNc2nnsc2C(F)F)C1 21657,O=C(C1CCCc2scnc21)N1CCCN(C(c2csnn2)=O)C(CO)C1 21658,CC1CCN(C(C2C(C(F)F)C2(C)C)=O)CCN1C(=O)CSc1ccccc1Cl 21659,C(=O)(C(C)CC(N)=O)N(CCCCN(C(C(C(C)O)N(C)C)=O)C)C 21660,C1(C(=O)NC2(CC=C)CN(C(=O)Cc3csc(Br)n3)C2)CC=C(C)CC1 21661,C(=O)(C1=CCCC1P(C)(C)=O)N(CCN(C(C(CCCC)CC)=O)C(C)C)C 21662,c1(OC)ccc(Br)cc1CC(=O)NC1CC2(C1)CC2NC(=O)CCCC#N 21663,CC1C2CC(C2NC(=O)CNC(c2ccccc2F)=O)N1C(c1ccc(Cl)s1)=O 21664,C(=O)(CS(=O)(=O)CC(F)(F)F)NC(C1CCN(C(c2c(OC)nn(C)c2)=O)C1)C 21665,Nc1cnc(Br)c(C(=O)NC2CCN(C(c3ccc(CO)cc3)=O)C2)c1 21666,c1(CNC(C2(C)CCCC2O)=O)nc(CNC(=O)C2=COCCC2)cc(O)n1 21667,C1(CNC(C2(CCC)CCNC2=O)=O)CN(C(C2(Cl)CC2)=O)CC12CCC2 21668,N(C1c2ccccc2OCC1C)C(c1ncnc2sc(C)c(C)c12)CC 21669,C(=O)(C(C)S(C)(=O)=O)N(CCCN(C(c1c(CCC)occ1)=O)C)C 21670,C1(C)(CC)C=C(C(=O)N2CC3CC(NC(c4cccc(=O)n4O)=O)C3C2)C1 21671,CCC(CC(=O)NCc1cn(C2CC2)nn1)NC(=O)C(O)Cn1cncn1 21672,CC1CC(NC(C2CCCN(CCNS(C)(=O)=O)C2)=O)CCS1 21673,N1(C(CCC)=O)CCCC(CNC(=O)Nc2[nH]cnc2CC)C1.C(C)(C)(C)NC(=O)O 21674,C1(C(=O)NC(C(C)C)(C)C)CC(=O)CN1C(=O)CCc1ccncc1 21675,C1(CNC(C=CCC)=O)CCC2CN(C(=O)CCC(=O)NC)CCC2C1 21676,c12cccc(c1)CO2.C(=O)(CP(C)(C)=O)NCC(CNC(c1nc(C)sc1)=O)F 21677,N1(S(=O)(=O)Cc2nnc(Cn3cc(Br)cn3)o2)CCCC(CN=[N+]=[N-])C1 21678,c1(NC(N2C(C)CC(CNC(=O)CNC=O)C2)=O)cc(Cl)ccc1OC(F)F 21679,c1(CC)ccc(CC(N2CCN(Cc3cc(-c4ccccc4)n[nH]3)CC2)=O)cc1 21680,C(C(C(=O)N1CCN(C(=O)C=C2CCSCC2)CC1)C(C)(C)C)OCC=C 21681,Cc1nn(C2CCC2)cc1C(=O)NC(C(C)NC(c1ccc(Cl)[nH]1)=O)C(C)C 21682,O=C(C(O)Cn1cncn1)NCCC1CCN(C(=O)CCOCC2CC2)C1 21683,Cc1cc(C(F)(F)F)nc(N2CCCOC(CNC(=O)CC3(CO)CC3)C2)n1 21684,CC1(C)CC(C(=O)NC2CCCCC2CNC(C2CCCN2S(C)(=O)=O)=O)=NO1 21685,N1(C(C(c2cnn(C)c2)NC(C=CCC)=O)=O)CCC(C)(O)C(O)C1 21686,c1(NC(CCC(CC)NC(=O)C(CC)C(F)(F)F)=O)cnn2cccnc12 21687,C1(CNC(CCC=CC)=O)CCC2CN(C(C3(C#N)CC3)=O)CC12 21688,N#CC12CC(C(=O)NCC(N3CCCC3CC(N3CC4CC3C4)=O)=O)(C1)C2 21689,c1(C(N2CC(C)C(NC(=O)CCC(C)(C)O)C2)=O)cc([N+](=O)[O-])n[nH]1 21690,Cc1ncc([N+](=O)[O-])cc1C(=O)NCC=CCNC(C1CC(C2CCCC2)C1)=O 21691,N1(C(C2C(CCC)CCC2)=O)CCSCC1CCNC(=O)Cn1nnnc1C 21692,C1(C)(COC)CC(NC(=O)C=CCNC(c2ccncc2Cl)=O)CCO1 21693,N1(C(Cc2cn(CC)nn2)=O)CCC(NC(=O)CC(C)C)C1c1ccccc1 21694,n1(CCOC)nc(C(N2CCC(C(C)NC(C3(CCO)CC3)=O)C2)=O)ccc1=O 21695,C=CCC(Cc1ccccc1)C(=O)N1CC(Cc2cc(OC)ns2)C1 21696,C1(CS(C)(=O)=O)CCCC1(c1nnnn1CCSC1CC1)OCCNCCF 21697,C1(CCC(=O)N(CC(C)(C)NC(C=C(C)C(C)(C)C)=O)C)CCCCN1C 21698,N1(C(COC(CCC)=O)=O)CC(CNC(=O)CCCOC(C)C)OC2COCC12 21699,c1(C(=O)NC2CCC(CNC(C3NC(=O)OC3)=O)C2)cccc(Cl)c1Br 21700,n1(C(C)C)cnc2c(N3CCC(C)=C(C)C3)[nH]c(=NCc3ccncc3N)nc12 21701,c1(C(N2CCN(C(c3c(OC)nccc3)=O)C(CO)C2)=O)nc(O)nc(O)c1N 21702,c1(OC)ccc(Cl)c(C(=O)NCC2CN(C(c3cnc(C4CC4)s3)=O)C2)c1 21703,N1(C(c2n(CC)ncc2)=O)CC2CCCC1(CNC(c1coc(Cl)c1)=O)C2 21704,C(c1ccccc1)=CCC(=O)NC(C)(C)CNC(=O)Cc1csnn1 21705,Cc1cc(CN2CCC(CCNC(=O)CCOc3ccccc3F)C2)ccc1Br 21706,C1(C(=O)NCC2CC(NC(C(n3ccc(C)n3)C)=O)C2)CCOC(C)(C)C1 21707,N1(C(c2nc(Cl)c(Cl)s2)=O)CC2CCN(C(c3ccnn3CCF)=O)C2C1 21708,C1(C(N2C(C(=O)NCC(CCC)O)CSC2)=O)CC(C)CCO1 21709,Cc1nc(Br)oc1C(=O)N(C1CCCC(NC(C2(CCF)CC2)=O)C1)C 21710,N1(C(C(=O)NCC)=O)CC2(C=C(C(=O)NC(C3CCN(C)C3)C)CO2)C1 21711,c1(OC)cc(C)c(C(=O)NC2CC3(C2)CC3NC(=O)CC2CCCN2C)cc1Cl 21712,C1(C(N(C)CCOCCNC(=O)C=CC2CCCC2)=O)CCCCC1C(F)(F)F 21713,Cc1ccnc(C(=O)NC2CC2CNC(c2snc(O)c2Cl)=O)c1N 21714,C(=O)(CC1OCCc2ccsc21)N1CCN(C(C(CC=C)N(C)C)=O)C(C)C1 21715,c1(C(=O)NCC2C(NC(C(COC)OC)=O)CC2)cc(=O)n(C)cc1Br 21716,CCC(C(=O)NCC1CCN(C(c2cnn(CCF)c2)=O)C1)C(C)(C)CC 21717,N1(C(CC(=C)I)=O)CCOCC(n2cc(C(C3CCOCC3)C)nn2)C1 21718,C(=O)(C(C)(F)C(C)(C)F)NCCCOCCN(C(c1cnc(C(C)C)nc1)=O)C 21719,C1(C(=O)NCC2CCCN(C(=O)Cc3ccon3)CC2)Cc2n[nH]cc2C(=O)N1 21720,CCC(CNC(=O)CCS(N)(=O)=O)(CC)C(=O)NCC1CCOC(C)(C)C1 21721,Cc1ccc(C(=O)NC(C)CN(C(=O)CC2COC(=O)N2)C)c2c1CCC2 21722,c1(NC(C2NCCN(C(C(C)O)=O)C2)=O)cc(F)c(Cl)c(Cl)c1 21723,c1(CC(=O)NC(C2CN(C(=O)C#CC3(C)CC3)C2)C)c(Br)ccc(F)c1F 21724,CCC(CC(F)F)C(=O)NC1CCN(C(=O)CCC2CC2)C1 21725,C=C(C)CCC(C)NC(c1cccc(Cn2cc(CNNS(C)(=O)=O)nn2)c1)=O 21726,c1(C(=O)NCC2C(C)(C)C(NC(C34CSC(C3)C4)=O)C2)ccc2c(c1)OCCO2 21727,N1(C(CCN(C(C)=O)C)=O)CC2CC(C1)CN(S(=O)(=O)c1ccc(F)cc1)C2 21728,C(CCNC(=O)C(C)CO)(C(=O)NCCCN1CC=CC1)OC 21729,c1(C(C(=O)OCC)=O)c[nH]c(=NCC2CCN(C(c3cncn3C)=O)C2)c(C)c1 21730,c1(CNCc2c(OC)nc(C)cc2)[nH]c2ccccc2c1Cl 21731,CCC(C)C(C(=O)N1CCC(C(F)(F)F)C(NC(=O)Cc2ccnn2C)C1)OC 21732,Cc1ccc(CNC(C2CSCCN2C(=O)CC2NC(=O)NC2=O)=O)nc1 21733,Cc1csc(=O)n1CC(=O)NC(C1CCCC1)CNC(=O)C(C)N=[N+]=[N-] 21734,C1(C2CCOCC2)(C(=O)NC2CC(NC(C34CCCC3C4Br)=O)C2)CC1 21735,c1(C(=O)NC(CC(C)NC(C2CCC(=O)N2)=O)C)ncccc1OC(F)F 21736,c1(OC)cc(F)cc(C(N2CCC(N(C)C(C3CC(CC(F)F)C3)=O)C2)=O)c1N 21737,C1(NC(C=CC(C)(C)SC)=O)CCCN(C(C2CCCCCO2)=O)C1 21738,S(=O)(=O)(c1ccc(C(N2C3CN(C(=O)C(C)(C)C)CC23)=O)cc1)N(C)C 21739,C(CO)(CCCCNC(c1ccc(=O)n(CC(C)O)c1)=O)NC(C(C)OCC)=O 21740,C1(NC(C)=O)CCN(C(=O)OC(C)(C)C)CC1CSc1ccncc1Cl 21741,n1(CC)cc(S(=O)(=O)N2CC3CC2CC3NC(=O)Cc2ccc(Cl)cc2Cl)cn1 21742,n1(CCCN(CCO)C(c2c(C)ccc(C)c2)=O)cnc2c1CCCC2 21743,N1(C(c2c(=N)cc[nH]c2)=O)CCCC(NC(c2ccsc2Br)=O)C(F)C1 21744,c1(C(=O)NC2CCCCC2c2ccc(O)cc2)csc2c1CCNC2 21745,CC(CC(F)(F)F)N=c1[nH]c(NC2CCSc3ccccc32)nc2ccsc12 21746,c1(C(=O)NCCC(CC)(C)NC(=O)CCC(C)(C)C)ccc(C#N)cn1 21747,c1(C(=O)NCC(CNC(CCc2c(C)nn(C)c2)=O)C)ccc2c(c1)CN(C)C2 21748,C=CCCCC(=O)NCC1(OC)CN(C(=O)C(C)NC(C2CCC2)=O)C1 21749,C1(NC(=O)Cc2ccc(C(F)F)cc2)CC2CN(C(C3C4COCC34)=O)CC2C1 21750,C1(CNC(C2N(CC)CCC2)=O)C2CCC1CN(C(C1CCC1)=O)C2 21751,c1(CC)ccc(C(N2CC3CC(NC(=O)C=Cc4cnn(C)c4)C2C3)=O)c(C)n1 21752,N1(C(CCC=CC)=O)CCC(F)(CNC(C2CCC3(CCC3)O2)=O)CC1 21753,N1(C(CNC(=O)OC)=O)CC(C)C(N=c2[nH]nc(C3CC3)s2)C(C)C1 21754,c1(C(C(C)NC(c2ccsc2Br)=O)NC(C=C(C)C)=O)ccccc1 21755,C(=O)(CC(C(=O)OCC)C(C)=O)NCC1CCN(C(C(=O)NCC)=O)C1 21756,S(=O)(=O)(c1cccs1)NCC(=O)NC1CC(F)(CNC(c2ccco2)=O)C1 21757,c1(C(N2CCC(NC(C(CC=C)C)=O)C(C)C2)=O)nc2ccccn2n1 21758,c1(N(C)CC)nnc2c(C(=O)NCc3nn[nH]n3)ccc(C(F)(F)F)n12 21759,C1(NC(C(F)=CCC)=O)CC2CC(C1)N(C(C1CC1[N+](=O)[O-])=O)C2 21760,C(=O)(CC(CC1CC1)NC(C1C2CCC(F)C12)=O)N(CCC#C)C 21761,N1(C(CCCC)=O)CCC2(CNC(=O)C(c3ccc(Cl)cc3)O)CCCCC12 21762,c1(OC(C)C)nc(NC(N2CC(C)CC2c2cccnc2)=O)ccc1Br 21763,C(C)(C(=O)NC1CCC1NC(=O)COCCCOC)OCC=C 21764,CN1CC(C)(C)CC1C(=O)N(C1CCCN(C(c2cnc(C#N)s2)=O)C1)C 21765,Cc1ccc(C(=O)NC2CCN(C(=O)CCc3cnn(C)n3)C(C)C2)c(O)c1 21766,c1(C(C(=O)NCC2C(NC(C(C)C)=O)CCC2)N(C)C)ccc(O)cc1 21767,Cc1c(C(=O)NCC2CCCC(NC(C34CCC(C3)C4)=O)C2)cnc2ccnn12 21768,C1(C(C)NC(=O)C(c2ccn(C)c2)C)CCCN(C(C2CCCC2O)=O)C1 21769,N1(CC(=O)NC2CC(CCC(=O)O)C2)C(=O)CNC1=O.C12C=CC(C1)CC(=O)N2 21770,N1(C(c2c(OC)cncc2)=O)CCC(CNC(C2CC2C)=O)C(O)C1 21771,c1(C(N2CC3(CN(C(=O)CN4CCS(=O)(=O)CC4)C3)C2)=O)cc(I)c(F)cc1Cl 21772,CC1CC(NC(c2ccc(C3CC3)nc2)=O)CN(C(c2cnc(S)n2C)=O)C1 21773,CCC(CC)C(C)C(=O)NC(C1(CNC(=O)CC2=CCOCC2)CC1)C 21774,c1(C(C)C)ccc(C(N2CCC(CF)(NC(=O)CC3CCCC3(F)F)C2)=O)cc1 21775,Cc1nc(CC(C)C)sc1C(=O)NCC1CN(C(C2OC(C)CC2C)=O)CCO1 21776,CC(C(O)C(=O)NC1CC(CCNC(=O)Cn2cnnn2)C1)c1ccccc1F 21777,CC1CC(NC(C2CCC2)=O)CCN1C(=O)C(=C1CCCCC1)F 21778,Cc1cc(C)n(-c2ccc(-c3nc(-c4ccc(OC(F)F)nc4)n(C)n3)nc2)n1 21779,C12(CNC(=O)CN3CCNC3=O)CCC1CCN2C(c1ccccc1Cl)=O 21780,C(C)(CC(C)C(F)F)(c1n(CCCSCC)nnn1)N.c12ccc(cc1)OC2.OC 21781,N1(C(C2=CCC(NC(c3nc(C(C)C)oc3)=O)C2)=O)CCCC(C)(C#N)C1 21782,C(C(C)CN=c1[nH]c(=NC(C)c2cnn(C)c2)[nH]c2ccsc12)OC 21783,N1(C(CCN(C(=O)C(C(C)O)N(C)C)CC)=O)CCCC(C)C1CO 21784,c1(C(=O)OCC)cc2cc(NCC3CCCC3N)ccc2s1 21785,c1(C(=O)OC)nccc2cc(-c3ccc(OC)c(C(=O)OC)c3)ccc12 21786,CC(C)CC(CNC(=O)CC(C)NC(c1ccccc1)=O)NC(C1CC(F)C1)=O 21787,N1(C(C(C=C)C)=O)CCOCC1CC(=O)N(C1CCNC1=O)C 21788,Cc1cc(N)ccc1C(=O)NC(C)(C)CCCCNC(=O)CC1CCCOC1 21789,N1(C(CCCC#C)=O)CCC(O)(CCNC(c2csc(COC)c2)=O)CC1 21790,CC1CN(C(c2ccc(C3CCC3)nc2)=O)CC1NC(C1(F)CCOC1)=O 21791,Cc1ccc(S(=O)(=O)N2C3CCN(CC3)C(=O)C2)s1.C(=O)(C1=CCCCO1)NC 21792,C(C(CC(F)(F)F)NC(=O)CN1C(=O)CCC1=O)NC(CC(C)c1ccco1)=O 21793,c1(C(=O)NCC2N(C(C=Cc3nnc(C(C)C)o3)=O)CC2)cc2scc(Cl)c2[nH]1 21794,c1(C(=O)NCCC2CC(NC(C3ON=C(C(C)C)C3)=O)C2)cncc2c[nH]nc12 21795,S(=O)(=O)(c1cccnc1NCCCc1nncs1)N(C1C(C)CCCC1)C 21796,C=CCCCCC(=O)NCC(C(C)C)NC(=O)CN1C(=O)CCCC1=O 21797,C1(C)(CNC(C(C)c2ccco2)=O)CCCC1NC(c1cnc(C(F)F)s1)=O 21798,C=CCC(C(=O)NCCCCN1CCN(C(=O)C(O)CCSC)CC1)NC(C)=O 21799,c1(-n2ncc(C(N3CC(C)(NC(CCOC)=O)C3)=O)c2)ccc(F)cc1 21800,c1(SCC(=O)NC2CC(Nc3cc(OC)nc(SC)n3)C2)nc2ccccc2s1 21801,CCC(C)(C)C(=O)C(=O)NC1CC(C)N(C(=O)C(C2CCCC2)OC)C1 21802,Cc1ncc(N)cc1C(N1CC(CNC(C2CCCCCN2C)=O)C(F)(F)C1)=O 21803,c1(SC)ccc([N+](=O)[O-])cc1C(=O)NCCCC(C)(C)NC(=O)CC1(CO)CC1 21804,CCCCC(CNC(c1c(C)nsc1N)=O)NC(=O)CCN(CC)CC 21805,c1(OC)ccc(OC)c(C(=O)NCC2CN(C(c3sncc3C)=O)CCO2)n1 21806,c1(C(=O)NC2(C)CC(NC(C=C(CC)CC)=O)C2)cccc(-n2cncn2)n1 21807,CC(C)S(=O)(=O)CC(=O)NCCCNC(c1nc(=O)n(C)[nH]1)=O 21808,c1(C(F)(F)F)cc(C2(CN(CCCO)CC3COC3)CC2)ccn1 21809,C(=O)(C(C(F)(F)F)C(F)(F)F)NC1(C2CN(C(c3ncc(CC)cn3)=O)C2)CC1 21810,N1(C(CCSCC)=O)CCN(C)CC1C(=O)NCc1nnn(C)n1 21811,c1(C(C)C)cc(N2CCCC2CNC(=O)CC(C)C2CC2)n2ncnc2n1 21812,CC1CC(NCC2CCN(C(C)(C)C)CC2CO)CC(C)O1 21813,C(=O)(CC(C)(C)CC(F)(F)F)NCCCNC(c1cnc(OC)nc1)=O 21814,C1(c2cccs2)(CSC2CC23CC3)CCCC1 21815,N1(C(C(C)OC2CCOC2)=O)CCCC1C(C)NC(c1ccc(F)s1)=O 21816,c1(CCC(=O)NCCCN(C(C(CCC)NC(C)=O)=O)CC)ccc(C)cc1C 21817,C1(CNC(C(C(C)C)NC(C)=O)=O)CCC2(CN(C(=O)C(C)C(C)(F)F)C2)O1 21818,c1(C(=O)NCC2C(CNC(C3C(C)(C(F)(F)F)C3)=O)C2)ccn2nccc2c1 21819,C=CCCC(CO)NC(c1nc(CNC(c2ccncc2)=O)oc1C)=O 21820,C1(NC(C2(CNC(C(C)N(C)C)=O)CCCO2)=O)CC2(C1)CC(O)C2 21821,c1(C(N2CC(F)C(F)C2)=O)ccc(CNCc2cccc(F)c2)c(Br)c1 21822,CCC(C(=O)NC(C(=O)NCC1C2COCC12)C1(O)CCC1)n1ccnc1 21823,C1(CN(C(C2C=CCCC2)=O)C2CC2)C2CN(C(=O)COCC(F)F)CC12 21824,C1(CNC(C2Cc3nccn3C2)=O)CC2(CCC2)CN1C(=O)Cn1ccnn1 21825,C(=O)(C#CC1CCCOC1)NCC1CN(C(C(C)N2CCC2)=O)CC1C(F)(F)F 21826,C1(NC(c2cc(Cl)ccn2)=O)CC2CC1N(C(=O)C(C1(O)CCCC1)F)C2 21827,C1(CC(=O)NCc2cccc(F)c2)CC2(C1)CN(C(=O)Cc1cnns1)C2 21828,C1(C(=O)OC(C(=O)OCC)Cc2ccc(F)cc2)CC(=O)N(CC(F)(F)F)C1 21829,c1(C(=O)NCCC2N(C(C3C(OCC)C3)=O)CCCC2)c2c(c[nH]c1=N)CCC2 21830,N1(C(=O)Cn2cncn2)CC2CN(C(C3(c4cccc(F)c4)CC3)=O)CC2C1 21831,C(c1cc2c(cc1OC)CC(C)O2)=CC(=O)NCCN(C(=O)C(F)F)CC 21832,c1(C(N(CCCNC(=O)CC(C)C(F)F)CC)=O)cn2cc(C)c(C)cc2n1 21833,C=CCC(C)(C)CC(=O)N1CCC(C)(C)C1C(=O)NC1CCNC(=O)C1 21834,C1COc2ccccc2O1.N12CCC1(CCO)C(n1cccn1)NC(=O)C2 21835,C1(C(=O)NC2(CCCC(=O)NC3CC4CCC3C4)CCC2)OC2CCC1C2 21836,C12(CC(=O)N(CCCCO)C)CCC1CN(C(C1(C(N)=O)CC1)=O)C2 21837,N1(C(c2c(CNC(C(C)CO)=O)ccs2)=O)CCC(C)C1c1ccccc1 21838,c1(NC(C(N2CCC(C(=O)OC)C2(C)C)=O)=O)ccc(N=[N+]=[N-])cc1 21839,CCCCC(O)CC(=O)NC1(COC)CN(C(c2ccc3c(c2)C(C)CO3)=O)C1 21840,N1(C(C(CC(C)C)=O)=O)CCC2(CC1)CC2CNC(=O)CCCc1cccs1 21841,C1(C(=O)NCC2CN(Cc3c(C)ncs3)C2)CC(=O)N(C)C1c1cccnc1 21842,C1(C(=O)NCc2c(C)cn(C)n2)CN(C(=O)C(CO)C(C)(C)C)CC1C1CC1 21843,n1(C(C)C(N2CC=CC(NC(=O)C(C)(F)F)C2)=O)c(S)nc2ccccc2c1=O 21844,N1(C(c2c(CC)nn[nH]2)=O)CC(C(N2CC(S(C)(=N)=O)C2)=O)OC(C)C1 21845,c1(C(N2CCC3(CNC(=O)O3)C2)C(=O)NCCC#N)cn2cc(Cl)ccc2n1 21846,c1(C(=O)NCCCN(C(C(C2CCOCC2)OC)=O)CCO)cn(C)[nH]c1=N 21847,c1(OC)cc(F)c(C(=O)N(CCCNC(c2cccc3c2COC3)=O)C)cc1N 21848,C1(C(=O)NC(CNC(c2sc(CC)c(C)c2)=O)(C)C2CC2)CC2CSCC(C1)C2 21849,C(=O)(CCN=c1[nH]c(=NCCC(C)C(F)F)c2sccc2[nH]1)NCC(C)C 21850,C(=O)(C1CCCn2ccnc21)N1CC2(C(NC(C(CC)OC)=O)CCC2)C1 21851,N1(C(CN(C(=O)CCc2cc(Cl)no2)C)=O)CCN(C(c2ccoc2)=O)C2CC12 21852,CCCC(C(=O)N(CC(CC)NC(c1ocnc1C(C)C)=O)C)C(C)C 21853,N1(C(=O)NCC2CCC(O)C2)CCC(n2ncnc2C(=O)O)CC1 21854,O=C(CS(=O)(=O)Cc1noc(-c2ccc(C(F)F)cc2)n1)Nc1ccc(F)cc1 21855,N1(C(CC(COC)COC)=O)CCCCC12CN(C(c1cc(O)ncn1)=O)C2 21856,c1(NC2(CF)CCN(C(C(C(C)C)N3CCCC3=O)=O)C2)ccc(C#N)nc1 21857,N(C(=NCCCCl)NC1CC(=O)N(CCN(C)C)C1)C(C#C)Cc1ccccc1 21858,Cc1nn(C)cc1CC(=O)NCCC1CSCCN1C(=O)CC(C)(C)C1CC1 21859,N1(C(C2C(C)(C)C2C#N)=O)CCC(NC(=O)CSCc2cccnc2)C(CO)C1 21860,C1(C(N(C)CC2(C)CCCO2)=O)C2CC1N(C(C1(CF)CC1)=O)C2 21861,c1(C(=O)NC2(N3CCCC3)CC2)cc2c(nn1)CCC2.C12CCC1CNC(=O)C2 21862,C1(n2cc(C(=O)NC3CCCC3)nn2)CCN(C(=O)Cc2csc(CO)n2)CC1 21863,C(=O)(C(C)(C(=O)OCC)OC(C)(C)C)N(C1CCCN(C(CSCC)=O)C1)CC 21864,C(=O)(C(c1cccs1)NC(=O)C(C)n1cccn1)N(CCF)CC 21865,c1(SC)nc(Cl)c(CN2CC(C(N3CCCCC3C)=O)CC(F)C2)c(Cl)n1 21866,N1(C(C(C)OCC)=O)CCCC(N(C(c2cc(SC)oc2C)=O)CC)C1 21867,N1(C(C2(OCC)CCOCC2)=O)CC(NC(c2cnccc2C)=O)CC(O)C1 21868,C(CC(C)C(=O)NCC1(C(=O)N(CC)Cc2cnc[nH]2)CC1)=CCC 21869,c1(N(C(C)=O)C)ccccc1C(=O)N(CC(C)CNC(=O)CC1OCCCO1)C 21870,C(C(C(C)(C)C)NC(c1cc(-c2ccoc2)[nH]n1)=O)NC(c1c(C)ocn1)=O 21871,N1(C(C(c2ccn(C)n2)C)=O)CCCCCC1C(=O)N(C)Cc1nccs1 21872,CC(C)CC(O)C(=O)N1CCCC(C(C)C(=O)NCCC#CCO)C1 21873,C(=O)(C(C)(O)CC(C)C)NCC(CNC(c1c(C)nc(Br)o1)=O)F 21874,N1(C(=O)NCC(=O)Nc2oc(C)c(C(=O)OC)c2C#N)CCS(=O)(=O)CC(C)C1 21875,c1(C(=O)NC(C)CCCCNC(C2CC3(CSC3)C2)=O)ccc([N+](=O)[O-])s1 21876,N1(C(C(C)CC2CCCC2)=O)CCCC(O)C1.C12(CC1)C(=O)N2 21877,C(=O)(CCC(=O)NC1(C)CCN(C(=O)C(C)OCc2ccncc2)C1)OCC 21878,c1(C(N2CCOCC2(C)C)C(=O)Nc2cccc(OC)c2)nnc2c(=O)[nH]ccn12 21879,c1(C(CNC(c2cccnc2)=O)OC)oc(Cc2ccc(N(C)C)cc2)cc1C 21880,c1(CC#N)ccccc1CC(=O)NC1C=CCN(C(c2ccc(Br)cn2)=O)C1 21881,CC(C(=O)NC1CC(NC(=O)C(C)N2CCC2)C1)S(C)(=O)=O 21882,c1(C(=O)NCC(CNC(C2(CCC)CC2)=O)C)cnc(C(C)(C)C)[nH]1 21883,C=CCCCCCCCC(=O)NCCOCCNC(=O)C(c1c(C)n[nH]c1C)C 21884,C=CC(C)(CC)C(=O)NCC1(F)CC(NC(=O)C(C)OC)C1 21885,CCC(CC(=O)NCCC1(O)CCN(C(=O)C(C(C)C)NC(C)=O)C1)OC 21886,c1(C(N2CC(CNC(c3cc(Br)no3)=O)C3C2C3)=O)ncc2ccccn12 21887,N1(C(CCNC(COC)=O)=O)CCCN(C(C2CC2[N+](=O)[O-])=O)CC1C 21888,C1(CC(=O)NCC2C3COCC23)(NC(=O)CC2CCOC2=O)CC(F)(F)C1 21889,O=C(O)CC1CCN(Cc2cn3ccsc3n2)c2ccccc21 21890,C(CCCC(=O)NCC1(OC)CCN(C(=O)Cn2ccc(C3CC3)n2)C1)OC 21891,CC1=C(C(=O)NCC2(C)CCC(NC(=O)Cc3cncn3C)C2)COCC1 21892,c1(-c2nc(NC(=O)Nc3scnc3Br)sc2)cccc(F)c1 21893,c1(CC(=O)NCC(C2CCC2)NC(c2cc(C)sc2)=O)ccc(Br)cn1 21894,c1(C(N2CC(CNC(c3cncc(F)c3)=O)C(O)C2)=O)coc2c1C(O)CCC2 21895,N1(C(CNC(=O)C=CC2CCC2)=O)CC2(CC2)CC1CO 21896,c1(C(N2CC(C(=O)Nc3cnc(Cl)cc3I)NCC2)=O)c(F)ccc(Cl)c1Cl 21897,c1(C(N2CC(NC(COCc3ccc(C)cc3)=O)C(F)C2)=O)cc(Br)c(C)cc1F 21898,C(=O)(CCCN=[N+]=[N-])N(CCC(C(C)C)NC(C1(C)CC=CCO1)=O)C 21899,Cc1cc(N2CCC(CNC(C3CCc4c[nH]nc4C3)=O)C2)n2nc(C)nc2n1 21900,N1(C(C2(CC)CC2)=O)CCCC2C1CCN2C(c1cn(CC(F)(F)F)cn1)=O 21901,Cc1cc(C(=O)N(C)CCC2CCN(C(=O)C(F)C(C)C)CC2)ccn1 21902,c1(OCC)ccc(C(=O)NCC2CC(NC(C34CCCN3CCC4)=O)C2)c(O)c1 21903,C(=O)(C(C(C)C)n1cccc1)NC(C1CCN(C(c2cc(OCC)no2)=O)C1)C 21904,c1(NCC(N2CCC=C(Br)C2)=O)ccc(-c2nn[nH]n2)cn1 21905,CCS(=O)c1ccccc1C(=O)NC1CC(NC(C2CC2C)=O)C1 21906,N1(C(C2(NC(=O)OC)CCCC2)=O)CC(C)N(C(=O)Cc2cc(C)on2)CC1C 21907,CCC(C)C(C)C(=O)NC1(C)N(C(CCCC2(C(=O)OC)CCC2)=O)CC=C1 21908,c1(CC)nc(C(=O)NCCC2CN(C(=O)C(C(C)OC)N(C)C)CCO2)c(N)s1 21909,c1(C(N(CC(CNC(CCCC=C)=O)C)C)=O)ccn2ncccc12 21910,C(CCC(C)(C)C(=O)N1CCC12CCCC2)NC(c1cnn(C(C)C)n1)=O 21911,c1(C(=O)NC(COC)C(N2CCC23CCCSC3)=O)c[nH]c2ncccc12 21912,CS(=O)(=NC(=O)c1ccc2n[nH]c(Br)c2c1)c1ccncc1 21913,C(CS(C)(=N)=O)NC(C(n1cc(CCC2CCOC2)nn1)C)=O 21914,O=C(C1=CCCOC1)N(C1C2CN(Cc3ccc(=O)oc3)CC12)Cc1ccccc1 21915,C1(CNC(c2ccc(NC)cc2)=O)CC(C(=O)N(C2(C3CC3)CC2)C)=NO1 21916,c1(CC)oc(C(=O)N(CC(C)NC(=O)C=Cc2ccsc2)CC)cc1C 21917,c1(CN2CCC(C)(C(=O)Nc3[nH]nc(OC)c3C#N)CC2)c(F)ccc(F)c1C 21918,Cc1cc(C(N2CCC(C(C)(C)NC(=O)CSCC(N)=O)C2)=O)cc(C)c1F 21919,c1(CN2C(CN(OC)CC3CC3)CC(C)C2)c(Cl)ccc(Cl)c1Cl.C1(C=O)C2COCC12 21920,CC(C)C(C(C)NC(c1cn(C(C)C)cn1)=O)NC(=O)CCC1CCC1 21921,CON(C)C(=O)C1(NC(=O)CCC2(NC(c3nccn3C)=O)CCC2)CC1 21922,C12(C(N(CCN(C(CCc3cc(C)on3)=O)C)C(C)C)=O)CCCC1CC2 21923,Cc1ccnc(C(=O)NC2CCN(C(=O)CN3CCCC3C)CC2CO)c1O 21924,CC1CCN(C(=O)C(N2CCC3CCOC3C2)=O)CCN1 21925,N1(C(C2CC(O)(CC#C)C2)=O)CCOC(CC(=O)NCC2COCC2O)C1 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21944,CC1CC(C(=O)NCC2(F)CN(C(c3c(F)cccc3Br)=O)C2)=NO1 21945,C1(NC(C(C)N(C(C(CC)n2cncn2)=O)CC)=O)CN(C)C2(CCC2)C1 21946,C1(CC(=O)NC(C(C)NC(CN(CCOC)C)=O)CO)CCC(=O)N1C 21947,C(C(=O)Nn1cnnc1C)OC(C(C(=O)OCC)C(C)C)=O 21948,C1(C2CCN(C(=O)CCCCCn3cnnn3)C2)(NC(c2c(C)coc2)=O)CC1 21949,N1(C(c2n(CCCC)ncc2)=O)CC2CC2(CNC(=O)C=CC(F)(F)F)C1 21950,C(C)(C(CC(=O)N1CC(OC)C(F)C1)NC(c1c[nH]nc1C1CC1)=O)OC 21951,c1(C(N2CCC(NC(C)C)C(C)C2)=O)ccc2c(c1)CCC(C)(C)O2 21952,N1(C(CCC=C(C)C)=O)Cc2[nH]nc(C(=O)NC3CN(C4CCC4)C3)c2C1 21953,c1(C(=O)NCC2(O)CCN(C(c3c(C(C)C)nn(C)c3)=O)C2)cc2n(n1)CCC2 21954,C1(CNC(c2c(CCCC)ocn2)=O)CC(F)(F)CN1c1nnc(C(=O)OC)s1 21955,C(=O)(CC(C)(C)COC)N(CC(C)(C)NC(C1C(CC)CCC1)=O)C 21956,c1(CN(CCOC)C(C2(CF)CC2)=O)cccc(CNC(c2coc(Br)c2)=O)c1 21957,N1(C(CN(C(=O)OC)C)=O)CC(NC(=O)CCC2CCN(C)CC2)CCC1C 21958,N1(C(Cc2cc(C)nn2C)=O)CC(NC(C2(n3cc(Cl)cn3)CC2)=O)CC(C)C1 21959,c1(N(C)C)cccc(C(N2CCCCC2CNC(=O)CCC2CCCO2)=O)c1 21960,C(=O)(NNc1nc(C)nc(Cl)c1C)c1cc(OC)cc2c1OCC2 21961,c1(C(=O)NCC(C)(C)O)n[nH]c2c1CCN(C(c1cccc(F)c1O)=O)C2 21962,C1(C)(NC(C(CCC)O)=O)CCN(C(=O)CCC2CC2(F)F)CC1 21963,c1(C(N2CCC(CNC(CN(CC)CC)=O)(OC)C2)=O)c(C)ccc(F)c1N 21964,Cc1cc(C(=O)Nc2ccc(Br)c(-c3nn[nH]n3)c2)nc(C2CC2)n1 21965,c1(C(=O)NCC2CCC(NC(c3cnnc(Cl)c3)=O)C2)ccc2nn[nH]c2n1 21966,C(=O)(CC(Cl)Cl)N(C)CC=CC(=O)N1CCC1 21967,N1(C(C2CC(C)OC2)=O)CC2CCC1(CNC(C1CCC=CCC1)=O)CC2 21968,c1(C(C(=O)NCC(CC2CC2)OC)NC(=O)C(C2CC2)SC)cccnc1 21969,N1(C(C(CC)C#N)=O)CCC2(C(=O)NC3(C)CC4CCC3C4)CCCC12 21970,N1(C(C2(COC)CCC2)=O)CCC(F)(CNC(=O)CCn2ccnn2)C1 21971,C1(C(=O)NC2CC(N(C(CCNC(C)=O)=O)C)C2)Cc2ccccc2S1 21972,N1(C(COCP(C)(C)=O)=O)CCN(C(c2ccc(Cl)s2)=O)CC(CO)C1 21973,Cc1cc(NCCN)n2ncc(C)c2n1.C1(C(C=O)C)CCCCC1 21974,CC1CC(NC(=O)CN2CC3CC3C2)CN(C(c2cc3sccc3s2)=O)C1 21975,c1(C(N2CC(NC(C3(F)CCCCC3)=O)C(O)C2)=O)ccc(Br)c(O)n1 21976,C1(C(N(CCCNC(Cc2n(C)ccn2)=O)C2CC2)=O)CC2CCCC2C1 21977,CN1CCC2(CCN(C(CCC3CC(F)(F)C3)C(=O)NC3CCCCC3)C2)C1 21978,N1(C(C=CC(C)C)=O)CCC2CC(NC(C3CC(=O)N3)=O)CCC2C1 21979,O=C(CCCCCNC(C1OCC2CCCC12)=O)NC1CC2(C1)CC(O)C2 21980,C(=O)(n1nccc1NC(c1ccc(O)c(C(F)(F)F)c1)=O)OC(C)(C)C 21981,C(=O)(C(O)CC(C)C)NCC1(COC)CN(C(=O)CCC2(C#N)CCC2)C1 21982,c1(C(=O)NC2CCN(C(C3CC(C)OC3)=O)CC2)cccc(Cl)c1 21983,c1(NC(C(CSCC)NC(c2ccnc(OC)n2)=O)=O)cc(Cl)cc(Cl)c1 21984,C1(NC(c2cc(C(C)C)ncc2)=O)CN(C(c2cnco2)=O)CC1C#N 21985,C1(C(=O)NCC2(OCC)CN(C(=O)C(C)Nc3ccccc3)C2)CCC(C)(C)O1 21986,C(CC(C(C)(C)C)NC(c1coc(Cl)c1)=O)N(C(=O)CC1CCOCC1)C 21987,C(=O)(C1=CCCOC1)N1CC(CCO)(NC(C2CCC(C)(CC)O2)=O)C1 21988,N1(C(c2c(OC)cc(OC)nc2)=O)CC2CC(C1)N(C(C1CCC3(CC3)C1)=O)C2 21989,CC1C(C(N2CCC(C3OCCCC3NC(=O)C3=NOCC3)CC2)=O)CCN1C 21990,N1(C(CC2COCC(C)O2)=O)CCN(C(c2ccccc2Cl)=O)C(CO)C1 21991,c1(CN(C(C2(OC)CCSC2)=O)C)cnn2c1CN(c1ccnc(CO)n1)CC2 21992,C(=O)(C1=NNC(=O)CC1)NC(C1(NC(=O)C(C)Cc2ccccc2F)CCC1)C 21993,CC1(C)CCCC(CC(N2CCC3(CC3NC(=O)CN3CC4CCC3C4)C2)=O)C1 21994,C(=O)(C(C(C)C)C1CCC1)NCC(NOCCCC=C)=O 21995,C1(NC(CNC(N)=O)=O)CCCCC1NC(=O)Cn1cc(CNC2CC2)nn1 21996,c1(CN(CCC)C(=O)NC2CCC2C)ccc(F)cc1 21997,CN1C(=O)C2CN(C(C3CC4CC4C3)C(=O)NCC(F)F)CC2C1=O 21998,c1(CNC(CC2C(C)(C)C2CN=[N+]=[N-])=O)ccc2c(c1)S(=O)(=O)C=C2 21999,c1(CCC(=O)N(CC(C)NC(C2CC(CF)C2)=O)C)ccccc1OC(F)F 22000,C1(CC=C)(NC(=O)CC(C)OC)CCN(C(=O)CSC(F)(F)F)C1 22001,Cc1cc(=NC(C)C2CCOCC2)[nH]cc1C#N 22002,c1(-c2cn(C)nc2)ccc(NC2CCOC(c3ccc(F)cc3)C2)cc1Cl 22003,N1(C(=O)CCC2CCC2)CCC2(CC1)CCN(C(C1(CC3CC3)CC1)=O)C2 22004,C(=O)(N=c1cc(C)n(C(C)C)[nH]1)C1(OC)CCN(C(=O)CC2CC=CCC2)C1 22005,N1(C(=O)NCCCOc2ccc(F)cc2)CCS(=O)CC1c1ccccc1 22006,C(=O)(CC(C)C(F)(F)F)NC(CC)CCC(=O)NCC1CC12CCCCC2 22007,CS(=O)(=O)c1csc(C(N2CC(NC(C3CCCO3)=O)C(C3CC3)C2)=O)c1 22008,c1(CC(=O)NCC2(OC)CN(C(=O)C(C)O)C2)ccc(-c2ccccc2)cc1 22009,C(C(C)C)(C(O)C(=O)NC(C)(CSC)C(=O)NC(c1cccc(C)n1)C)OC 22010,C1(O)(C(c2ccccc2)NC(N2CC(C(=O)OC)(CO)C2)=O)CCOCC1 22011,N1(C(C(C)c2ccsn2)=O)CCC(CCNC(C2CCCC2)=O)C(F)(F)CC1 22012,C(=O)(C(CCNC(=O)C(C)c1cc[nH]n1)OC)NCC(C#C)CC 22013,C1(C(N(CC(C)(C)NC(C(C)SC)=O)C)=O)CCNC(=O)C1 22014,CN=c1nc(C(N2CCN(C(=O)C#CC3CC3)C(C)C2C)=O)cc(C)[nH]1 22015,C1(C(=O)NC(CN(CCOCCC(C)C)C)C)CN(C)CCO1 22016,c1(C(=O)NC(CNC(c2cncc(OCC)c2)=O)CO)ccc(OC)c(OC)c1 22017,C1(NC(C2(C)CCCC2)=O)CCOC(C(=O)NC(C2CCCCC2)CO)C1 22018,N1(C(=O)OCC)c2ccccc2CCC1C(=O)NCC(C1CCC(C)CC1)(C)O 22019,C1(NC(C2C(C=C)C2)=O)CCC(C)N(C(c2cc(-c3ccccc3F)[nH]n2)=O)C1 22020,Cc1cc(C(=O)NC(C)CCNC(c2c(C)noc2N)=O)nc(O)c1 22021,C1(NC(C2C3C(NC(c4cnc(CC)o4)=O)C4C(C3)C42)=O)C(C)(C)C(O)C1(C)C 22022,C(CC(=O)N(CCNC(C1(n2ccnn2)CC1)=O)C1CC1)=CCC 22023,c1(C(=O)NCCC(C)N(C(C2C(CC)OCC2)=O)C)c[nH]cc(Cl)c1=O 22024,Fc1cc(NCC(F)(F)F)cc(Cl)c1.c12c(C(F)(F)F)nn(c1Cl)C2 22025,N1(Cc2ccn(CC)c(=O)c2)CCC2(CCN(C(=O)CC(C)C(=O)OC)C2)C1 22026,c1(OC)cc(C2(C(=O)NCCCC(C)NC(=O)C(C)SC)CCCC2)ccc1C 22027,c1(C(N(CC#C)CCC)=O)cc2ccsc2[nH]1 22028,N1(C(C2C(C)(C)C2)=O)CC2CCC(NC(c3ncoc3C3CC3)=O)C2C1 22029,C(C1=CCN(C(=O)C(O)CC2CCCCC2)CC1)NC(CNC(N)=O)=O 22030,C12(O)CCN(C1)C2=O.c1(OC)ccc(C(=O)N(CC(C)C(=O)OC(C)(C)C)C)s1 22031,C1(CC(=O)NCC(CNC(c2oc(CC)c(C)c2)=O)C)CCc2ccccc2C1 22032,C1(CNC(COC)=O)CC2CCC1N2C(=O)Cc1ccc(OC)c(O)c1 22033,c1(C(C)NC(C(c2conc2C)N(CCC)CC2CC(F)(F)C2)=O)ccccc1 22034,c1(CC(=O)N(CCC)CCNC(=O)CC2CC2(Cl)Cl)ccnc(Cl)c1F 22035,C1(CCCN(C)C)CCCN(c2nnc(-c3ccccc3Cl)n2CCC#N)C1 22036,N1(C(C(C)(C)OC)=O)CCN(C(c2ccc(F)cc2Cl)=O)C(C(C)C)C1 22037,Cc1ccc(C(=O)NCC2(NC(C3CC(F)(F)C3)=O)CCOC2)nc1O 22038,N1(C(CC(=O)NCC)=O)CCN(C(c2c[nH]c(=N)o2)=O)C(CC(F)F)C1 22039,CCC(CCC(=O)NC1(CNC(c2ccc(CC)c(O)c2)=O)CCC1)OC(C)=O 22040,N1(C(c2ncc(CC)cn2)=O)CCCC(O)(CNC(C2CCCC(=O)N2C)=O)C1 22041,N1(CC(=O)NCC(C)N(C(c2ccc(Cl)cc2)C(N)=O)C)CCCCCC1 22042,N1(C(C2C(C(=O)O)C23CC3(F)F)=O)CCc2c(I)n[nH]c2C1 22043,N1(C(CCCCOC)=O)C2CCC1CC(CNC(=O)CC1CC(C)=NO1)C2 22044,CCC(C)C(C(=O)NCC(F)F)N(C)C.C1(=O)C(=O)NCCN1C.C(COC)S 22045,C1(C(=O)NC2(CC=C)CCC2)CCN(C(=O)C2CCCN2C(C2CCCC2)=O)O1 22046,c1(C(=O)OCC(=O)NCC2C(C(=O)OC)CCC2)cc(C)cc(C)c1 22047,C(C(C)N=c1[nH]c(=NCC2CC(=O)N(CC(C)C)C2)c2sccc2[nH]1)OCC 22048,CC(CC(C)(F)F)C(=O)NC1(C)CCN(C(=O)Cc2csc(-c3ccoc3)n2)C1 22049,CN1CCC2(CC1)CN(C(C1CCN(C(C3(C)CC=CC3)=O)CC1(C)C)=O)C2 22050,c1(C(N2CC(NC(c3cc(-c4ccccc4)on3)=O)C2)=O)csc(O)n1 22051,C1(C2(O)CN(C(C3(C)C=CCC3)=O)C2)(CNC(c2csc(C)c2C)=O)CC1 22052,c1(OC)cc(Br)cc(C(N2CCN(C(C3CC3F)=O)C(C(C)C)C2)=O)c1OC 22053,N1(C(C(C)Cc2ccc(Cl)cc2)=O)CC2CCC(C1)N2Cc1ccc(F)nc1 22054,c1(NC(CNC(C2(SC)CC2)=O)C(C)C(C)C)ncc(Cl)cc1[N+](=O)[O-] 22055,CS(=O)(=O)c1ccc(S(=O)(=O)N2CCOC3(CCC(NC(=O)CN)CC3)C2)cc1 22056,N1(C(c2ccc(C)nc2)=O)CCC(C2CN(C(c3c[nH]cc(Cl)c3=O)=O)C2)CC1 22057,CCN=C(NCC1CCCCO1)NC1CC(=O)N(C(C)(C)C)C1 22058,N1(C(CCOC(CC(C)C)C)=O)CCC(C2(NC(=O)CN(C)C(N)=O)CC2)C1 22059,c1(CSC)cnn2c1CN(C(c1cc(-c3cccc(C)c3)no1)=O)CC2 22060,C1(C(=O)NCCCNC(CC(OCC)OCC)=O)CC(=O)N(C2CC2)C1 22061,c1(C(=O)NCCC(C)NC(c2ccc(C)c(F)c2)=O)ccc2c(n1)OCCO2 22062,c1(CC(=O)NCC(C)NC(C2(CC)CCC(O)CC2)=O)c(C)nc2ccccn12 22063,C1(C(=O)NCCCN(C(c2c(C)cc(C)cc2C)=O)CC)CCCCC12CCC2 22064,C1(C(=O)NC(CC)C)CC(=O)CN1C(=O)C(c1ccccc1)F 22065,C(CCCCC(=O)N(C1CCC(NC(C2CCCC(C#N)C2)=O)CC1)C)OCC 22066,c1(CCNC(C(C2CCC2)NC(c2cc(Cl)n[nH]2)=O)=O)ccncc1F 22067,C(=O)(C(F)CCC(C)C)N1CCCC(C(N(CC=C)CCOC)=O)(CC)C1 22068,Cc1ccc(OCC(=O)N(C(C)CCNC(=O)C(O)C2CCCC2)C)cc1 22069,c1(C(=O)NCC(C)CN(C)C(c2cc(F)c(N)cc2F)=O)cnc2[nH]cncc1-2 22070,C1(C(C)(C)O)CCCN(C(=O)C(N2CCNCC2)C2CC2)C1 22071,C(=O)(CC(C)(C)C(C)(F)F)Oc1nc(C2CCN(C(C)=O)CC2)sc1 22072,c1(CNC(c2sc3n(C)nc(C)c3c2)=O)cc(Br)c2ccccc2c1 22073,c1(C(c2n(CC)nnn2)NC2CCCCC2SC)ccc(Cl)c(Cl)c1C 22074,Cc1cc(C)c(C(=O)NCC2CCCCN2C(=O)Cn2ncn(C)c2=O)c(C)c1 22075,N1(C(C2N(C(C(C)=CC3CC3)=O)CCN(C)C2)=O)CCC2CCC(C1)N2C 22076,CCCC(C)(C)C(=O)NC(C1CCN(C(=O)CNS(=O)(=O)N(C)C)C1)C 22077,C1(Cc2nc(C)sc2)CCN(N2CCOCC3(CC3)C2)C1 22078,N#CC12CCC(C(=O)NCCC3CCN(C(=O)CNc4nccs4)C3)(CC1)CC2 22079,N1(C(CN2CC(CC)C2)=O)CC2CC2(NC(=O)Cc2cncc(O)c2)C1 22080,N1(C(CCc2cc(C)[nH]n2)=O)CCCCC1CC(=O)NC(c1csnn1)C 22081,Cc1cnccc1C(=O)NC(C1CN(CC2CCC(C)O2)C1)C 22082,c1(C(=O)NCC23C(CN(C(C(CSC)C)=O)C2)C3)cccc(=O)n1C 22083,C1(CNC(C2CC3CCC2O3)=O)C2CN(C(c3ccc(-c4cccs4)o3)=O)CC12 22084,Cc1cc(C(=O)NC(C)(CNC(=O)C2=CCC2)C2CC2)nn1C(C)C 22085,CCC1=NOC(C(=O)NC(CCC2CC2)C(=O)Nc2ccccc2OC)C1 22086,C1(CNC(C(C)SC(F)(F)F)=O)CCN(C(=O)CCS(N)(=O)=O)C1(C)C 22087,Cc1ccc2c(N3CC4CC3C4)nc(=NC3CCCCCC3C)[nH]c2c1 22088,C1(CC(=O)N(CCNC(c2c(C)cco2)=O)C)CCCCN1C 22089,C(=O)(C(C(C)C)n1cnnn1)NCC1CCN(C(CN(C(C)=O)C)=O)C1 22090,CC(C)(C(=O)N1CC(C2CN(C(=O)Cc3ccon3)C2)C1)C1=CCSCC1 22091,C#CCC(C(=O)N(CCCO)CC#C)NC(c1cccnc1)=O 22092,C1(C(=O)NCC(C)C2CCC2)CCN(C(c2c[nH]c(=O)cn2)=O)C1(C)C 22093,C1(C)(C(N2CC3N(C(CSCC(=O)OC)=O)C(CC3)C2)=O)CC(C(C)(C)C)=NO1 22094,Cc1cccc(C(=O)N(CC(O)CNC(=O)C(C)SCc2ccccc2)C)n1 22095,N1(C(C2CC3(CCN(C(C(C=C)C)=O)C3)C2)=O)CCCC2(CCCC2)C1 22096,C(=O)(C1=CN=C2N=CNN2C1)N(C)CC1CCCN1C(c1[nH]ncc1C#N)=O 22097,Cc1nn(C)c(Cl)c1C(=O)NCC(C1CCOC1)NC(c1c[nH]c(Br)c1)=O 22098,C1(N(C(C=C(CC)CC)=O)C)CCN(C(C2CC(c3cccc(F)c3)C2)=O)CC1 22099,Cc1cncc(C)c1C(=O)NC1CC(C(F)C(N2CC3CC3(CO)C2)=O)C1 22100,C(=O)(C(CC(C)C)N(C)C)NCC(CCC)NC(=O)CCc1ccc[nH]1 22101,N1(C(C(CNC(CSCCC)=O)CC(C)C)=O)CC(C)OC(C)(C)C1C 22102,c1(NC2CC=C(C)CC2)ccc(S(=O)(=O)N2CCCCC2C(C)C)cn1 22103,N1(C(COC)=O)CC2CC(NC(c3ccc(NC(c4cccs4)=O)cc3)=O)C1C2 22104,N1(C(c2c(C)c(F)ccc2Cl)=O)CC2CC3CC2C1C3NC(c1ccccc1)=O 22105,Cc1ccn2ncc(C(=O)NC3CC(C)N(C(=O)CCCc4ccsc4)C3)c2c1 22106,c1(CCNC(c2cccc(NC(=O)NC)c2)=O)c[nH]c2cc(F)c(Cl)cc12 22107,CCC(C)(CNC(c1ccnc(C)c1C)=O)C(=O)NC1(CCF)CCC1 22108,N1(C(=O)NC)CCN(C(C2CC(NC(c3ccc(F)s3)=O)C(O)C2)=O)CC1 22109,CC1CC2(CCN(C(=O)CC3CCCC3)CC2)CN1C(=O)CCCCC(C)(C)C 22110,Cc1cnn(C(C)C(=O)NC2CCC2NC(c2ccn(C3CC3)n2)=O)c1 22111,C1(O)(CC=C)CCN(C(c2conc2CNC(C2CC(=O)C2)=O)=O)CC1 22112,c1(CN2CCC(O)(C(=O)Nc3cc(O)nc(O)n3)C2)ccc([N+](=O)[O-])cc1O 22113,n1(C(C)C)cnc(C(=O)NC(c2ccnn2C)C(=O)NCC2(C)CC2(C)C)n1 22114,c1(C(N2CC(O)(CNC(C3CCOC3=O)=O)C2)=O)coc2c1CCCC2 22115,C1(C(C)C(=O)NCCCc2ccsc2)CCN(C(c2scnc2Cl)=O)CC1 22116,CN1CCC2CN(C(=O)NCc3cc4c(s3)CCC4)CCC12 22117,C(=O)(CCCC(=O)N1CCN(C(=O)CC2CCCSC2)C(C2CCC2)C1)N(C)C 22118,C12COCCC1NC2c1nnnn1C1CC1.n1(CC)ccnc1C(=O)OCC 22119,c1(CSCCC)ccc(C(=O)NC2(CNC(C3CCOC3)=O)CCOC2)o1 22120,c1(CC(=O)NC(CC=C)CNC(C2(C(F)F)CCCO2)=O)ccc(F)cc1 22121,Cc1oc(C(C)(C)C)cc1C(N1CC(CNC(=O)C(O)CC2CCCCC2)C1)=O 22122,c1(N2CCC(C(=O)OCC)(NC(=O)OC(C)(C)C)C2)c(Cl)cc(SC)cc1Cl 22123,C1(CSC)C(=O)Nc2noc1n2.c1(OC)ccccc1 22124,C(=O)(CCS(=O)(=O)N1CCOCC1)N1C(CNC(C2(CCC)CC2)=O)CC1 22125,C(=O)(CC(C)C1CC1)NC(CN(C(=O)C(C)(C)OCC(F)(F)F)CC)C 22126,c1(C(=O)NC2CN(C(C3CCCN(C)C3)=O)CC(F)C2)c(O)ccc(F)c1F 22127,C(c1c(C)coc1C)=CC(N1CC(O)(C(C)NC(C=C(C)C2CC2)=O)C1)=O 22128,Cc1ncccc1C=CC(=O)NC1(CCCNC(c2nccn2C)=O)CC1 22129,c1(NC(C)Cc2nncn2C)[nH]c(=NCCc2ccncc2Br)nc2scnc12 22130,N1(C(C2C(C)(C)CC2)=O)CC2CCC1C1CN(C(c3c[nH]nc3[N+](=O)[O-])=O)CC21 22131,C(C(C(=O)NCC1CCOC1)N1CCC2CCC12)(C1CCCCC1)OCC 22132,c1(OCC)c(C(N2CCC(NC(=O)Cc3ccc(C)c(Cl)c3)C2)=O)cccc1F 22133,C1(CCC(=O)NCC(c2nnc(O)o2)(C)C)(NC(=O)C(=O)NC2CC2)CCCC1 22134,CC(=O)C(C)CC(C)C(=O)N1CCC(C)(C)CC1C(=O)N(CC(C)C)C 22135,c1(CN2CCC(CC(N3CC4CC4C3)=O)CC2)cccc2ccncc12 22136,C1(CNC(=O)CCN2CCC2)CCN(C(C23CC(C(F)F)(C2)C3)=O)CC1 22137,CN1CCOC(CN(C2CC2(C)C)CCCNC(=O)OC(C)(C)C)C1=O 22138,Cc1cccc(C)c1C(N1CCC(C)C(CC(N2CCSC(C)(C)C2)=O)C1)=O 22139,c1(CCOC)nc(=NCC2CN(C(=O)CC(O)CN(C)C)CCO2)s[nH]1 22140,C(C(C)(C)CC(=O)N(C1CC(C(N2CC3CCC3(C)C2)=O)C1)C)OC 22141,c1(OC)cc(Br)c(CCNC(=O)C(N)CCc2ccccn2)cc1OC 22142,C1(CC=C)(NC(c2cnc(C(F)F)s2)=O)CN(C(c2cc(C(F)F)cs2)=O)C1 22143,Cc1cc(C)c(CN2CCC(N(C(=O)C(C)C)C)C2)cc1C 22144,c1(CC)ncc(C(=O)NC2CCCN(C(=O)CCC(F)(F)F)C2CC)c(C)n1 22145,c1(CCC)onc(CN(C)Cc2cccs2)c1CC 22146,C1(NC(=O)CC(F)F)CC2CC1CN(C(c1cnnc(O)c1)=O)C2 22147,Cc1cccc2c1CCC2NC(c1cnc2n1CCC2)c1nnnn1C 22148,N1(C(CCC=C=C)=O)CC2CCC(C1)N(C(c1cc(CC)ccc1OC)=O)C2 22149,CC(C)CC(CNC(=O)CC1CCC(=O)C1C)C(=O)NCC(C)N(C)C 22150,Cc1cc(C(=O)N(C)Cc2ccncc2F)nn1C(F)F 22151,c1(C(N2CC(N(C(C3CN(CC(C)C)C3)=O)C)C2)=O)ccc2c(O)ncnc2c1 22152,N1(C(c2[nH]cc(C)c2C)=O)CCN(C(C23CCCC2C3(F)F)=O)CC(O)C1 22153,c1(C(=O)NCCCCC2CN(C(C(C(C)O)(F)F)=O)C2)cc2ccsc2n1C 22154,c1(CNC(C(C)N(CC)CC)=O)ncoc1C1CN(C(C2CCCS2)=O)C1 22155,N1(C(c2nc(C)[nH]n2)=O)CCC2(CCN(C(C3CCC(C4CCCO4)O3)=O)C2)C1 22156,C=C(Cl)CCC(=O)NCC1CCN1C(c1ccnn1CCCC)=O 22157,C(=O)(C1CCc2nccn21)NC(C)C(=O)NOC1CCCCCC1 22158,C(CC(C(=O)NCC1(O)CCN(C)C1)NC(=O)C(COC)CC)OCC 22159,C1(CC)CN(C(c2ccc(C#N)cc2)C(=O)NCC(F)F)CC2(CCCOC2)O1 22160,C12(NC(C(C)=CC3CC3)=O)CCC1CN(C(c1ccsc1C)=O)C2 22161,Cc1cc(NCCCCC(C)NC(c2c(F)cccc2F)=O)n2nc(C)nc2n1 22162,C(=O)(CS(=O)(=O)N1CCOCC1)NCC(C)CNC(C1(F)CCCC1)=O 22163,c1(N2CCOCC(C(N3CC4CC3CO4)=O)C2)ncc2[nH]ncc2n1 22164,c1(C(CC)NC(=O)C(=O)Nc2cnn(-c3ncccn3)c2)ccc(Cl)cc1 22165,CC1CCC(NC(=O)Cc2cn[nH]c2)CN1C(c1ccc(O)nc1Cl)=O 22166,Cc1cc(NC(C23CC2CN(C(c2ccno2)=O)C3)=O)c(F)c(Br)c1 22167,C1(NC(C2C(=C)C2)=O)COC2(C1)CN(C(c1cccc3nncn13)=O)C2 22168,N1CCC(OC2CCC2)C(CC)C1.c1(OCC)cc(C=O)oc(=O)c1 22169,C1(C(=O)NCC(CNC(c2ccn(CC(C)C)n2)=O)(C)F)CCCCC(=O)N1 22170,c1(CNC2CCC(C(=O)NCc3ccn(C)n3)CC2)c(Br)ccc(Cl)c1F 22171,N1(Cc2cc(Cl)c(Br)nc2)CCC2(CCSCC2)C1 22172,c1(CNC(C2(NC)CC2(C)C)=O)cc(Br)ccc1Cl 22173,C(=O)(CS(=O)CCC(F)(F)F)N1C2(CNC(CC=CCC)=O)CCC1CC2 22174,c1(C2C(C(=O)NC(CCC(=O)NC(C)(C)CC(=O)O)=O)C2)c(F)cccc1F 22175,N1(C(CCCC)=O)CCC2CCCC12C(=O)NCCCc1cnn[nH]1 22176,c1(C(=O)NCC2CC(C)N(C(=O)CC3CCC4CC4C3)C2)cnc2occc2c1 22177,C1(C(N(CCCNC(c2c(OC)nsc2)=O)C2CC2)=O)CCSC(C)C1 22178,Cc1cnc(C(N2CCCC(CN(C)CCc3cnn(C)c3)C2)=O)cn1 22179,c1(C(N(C)C2CC2)=O)ccc(NC(C2CCCN2C(=O)C2CC2)=O)cc1 22180,C(C)(C(=O)N1CCC(N(CCO)C(C2CC(C)C2)=O)CC1)(C(C)C)OC 22181,C(CCN=c1cccc(S(=O)(=O)N(C)Cc2cccc(F)c2F)[nH]1)OC(C)C 22182,C(=O)(CCCCC(F)F)N1CC(CNC(C2(C(C)(C)O)CCC2)=O)OCC1 22183,C(=O)(C1=CCCOCC1)N1CC(CC)N(C(c2cc(C)c(C)nn2)=O)CC1 22184,Cc1cc(C)c(CNC(=O)C(c2ccoc2)NC(c2cccc(O)n2)=O)cn1 22185,c1(C(N2CC(CNC(c3c(CCC)n[nH]c3)=O)(COC)C2)=O)c(C)nnn1CC 22186,C1(N(C(C2(SCC)CC(O)C2)=O)C)CC2CCC(C1)N2C(=O)CCCCN(C)C 22187,N1(C(CCC2C(=O)NC(=O)N2)=O)CCC(NC(c2cnccn2)=O)C2CC12 22188,C1(C(=O)NCC(C)N(C(c2cc(C)n(C)c2C)=O)C)CN(C)CCN(C)C1 22189,N1(C(c2c(C)snc2)=O)CCC(NC(=O)CC(C)c2cccnc2)C(F)(F)CC1 22190,C1(C(=O)Nc2ccc(OC)cc2)CCCCC1(C)NC(=O)CCOC1CCCC1 22191,c1(CNS(CCCC)(=O)=O)cc(NC(=O)CC(C)C(=O)OC)ccc1C 22192,C#Cc1ccc(C(N2CCCC(NS(C)(=O)=O)C2)C(=O)NCC(=C)C)cc1OC 22193,c1(C(C)C)conc1Cc1nn[nH]n1.C12CC(C1)CC(=O)N2 22194,N1(C(C2C3CN(C(CCC(C)OCC)=O)CC32)=O)CCCC12CCCC2 22195,Cc1ccc(C2C(=O)N2)cc1.C(=O)(CCCC1CC1)NCC(O)CNC(N)=O.O 22196,c1(C(N2CCC3(C(NC(C4N(CC)CC4)=O)C3)C2)=O)ccc2nonc2c1 22197,N1(C(C2C=C(C)CS2)=O)CC(F)CC1C(=O)NOCCCO 22198,C1(N(CC#C)C(c2cc(COC)cs2)=O)CCN(C(c2ccn(C)n2)=O)CC1 22199,c1(NC(C)=O)cccc(CN2CCN(Cc3nc(-c4ccco4)no3)CC2)c1 22200,C1(C(=O)NCCN(c2ccccc2)C(CNS(C)(=O)=O)=O)CCC(F)C1 22201,C1(Nc2ccc(COC(C3CCOCC3)=O)cc2)CCC2CC1CN2 22202,c1(CC(=O)NC2CCN(C(=O)C(=O)NCC3CC3)CC2)ccc2c(c1)CC2 22203,c1(C(N(C2CCN(C(c3ccn(C4CC4)n3)=O)C2)CC)=O)cc(OC)ncn1 22204,c1(C(N2C(C)C(C)N(C(=O)CN3CC4CC4C3)CC2)=O)cccc2c1CCC2=O 22205,c1(C(=O)NC2(C(N3CC(C)(CC=C)C3)=O)CCCCC2)cnc(C)c(C#N)c1 22206,N1(C(CCc2ccc(C)s2)=O)CCN(C(=O)C=Cc2cocn2)C(C)C1C 22207,C(=O)(C(C)CCCC(C)C)N1C(CCNC(=O)C=C(C)C)CC(OC)C1 22208,c1(SCCO)cc(=NC(=O)CCN(C(C2C(C)C2)=O)C2CC2)[nH]n1C 22209,C1(NC(c2ccnc(C)c2N)=O)CN(C(=O)CCCF)C2(CCCCCC2)C1 22210,c1(C(=O)NC(C(C)C)CCNC(=O)CC2NC(=O)NC2=O)ccc2[nH]ccc2n1 22211,N1(C(C(CC)N(CC)CC)=O)CC2(C1)CN(C(C1(C(F)F)CCCC1)=O)C2 22212,C1(C(=O)NCC(O)CNC(=O)Cn2ccnc2)(SC)CCOCC1 22213,c1(C(N2C3CN(C(CC(CCCC)O)=O)C(CC3)C2)=O)cc2sc(C)c(C)c2[nH]1 22214,C1(C(N2CC(F)CC(OC)C2)=O)CCN(C(C2CN(C(C)C)C2)=O)C(C)(C)C1 22215,c1(C(=O)OC)cnc(C(N2CCC(CC(=O)NC(C3CCOCC3)C)C2)=O)cn1 22216,N1(C(C2CCN(C)C2=O)=O)C2CCC1CN(C(=O)CC(C)(C)c1ccccc1)C2 22217,C12(C(CO)NC(C3C(NC(c4c(C)nc(Cl)s4)=O)C3)=O)CC3CC(CC(C3)C1)C2 22218,CCCCCC(C)CC(=O)NCC1C2CN(C(=O)C(c3ccc(C)o3)C)CC12 22219,CN1CCOc2cc(C(N3CC4CCC3CN(c3ccnc(C5CC5)n3)C4)=O)ccc21 22220,N1(C(CC2CN(C(C)=O)C2)=O)CCC2(CC(NC(=O)CCc3ccn(C)n3)C2)C1 22221,CC1OCCCC1C(=O)NC(C)CNC(c1cccc(OC(C)(C)C)c1)=O 22222,C1(O)(CNC(C=NOC)=O)CCN(C(c2csnc2C)=O)C1 22223,C1(C)(C(=O)NC2CCC(N(C)C)C2)CCN(C(c2csc(F)c2)=O)CC1 22224,N1(C(CC2(C=C)CCC2)=O)CC(CNC(C2CCC(=O)NC2)=O)CC(C)(C)C1 22225,C(C(CNC(C1C(C)C1C)=O)CO)NC(CC1(OC)CC1)=O 22226,CC1c2cc(C(=O)NCCCCC3CN(C(c4ncn(C)n4)=O)C3)ccc2OC1C 22227,C(=O)(C(CNC(=O)CCC(C)C)C(C)(C)C)N1CCCC(OC)C1 22228,C1(NC(CCC(=C)C)=O)CC(NC(c2ccc(S(C)(=O)=O)o2)=O)C12CCOCC2 22229,c1(CN2CC(F)(C(=O)NCCc3ccc(OC)cc3)C2)cc(F)cc(Br)c1Cl 22230,C(=O)(CC(F)(F)C(F)F)N1CCC(C)(CNC(=O)C(F)C2CCCC2)C1 22231,N1(C(c2c(SC)csc2)=O)CC2CCCC2(NC(C2OCCC2(C)C)=O)C1 22232,N1(C(c2ccc(SCC)nc2)=O)CCC(OC)C(C)C1 22233,Cc1cn(C(C)(C)C(=O)NCC(=C2CN(C(c3cc(C(N)=O)[nH]n3)=O)C2)F)cn1 22234,C(C(=O)NC1CCC(NC(C2(N3CCCC3)CC2)=O)CC1)(C(C)(C)C)NC(C)=O 22235,C1(CNC(C(CCC)OC)=O)CC2(CCOCC2)CN1C(=O)CSSC 22236,S(=O)(=O)(CC(=O)NC1(C)CC(C(=O)NC2CC23CCC3)C1)NCC 22237,N1(C(C(C)NC(=O)NC)=O)CCN(C(=O)C(C)=C(C)C)CC1CC1CC1 22238,Cc1cc(C(N2CCOCC2CS(C)(=O)=O)=O)ccc1C#N 22239,N1(C(c2ccc(Oc3ccccn3)cc2)=O)CC(CO)C2(CCOCC2)C1 22240,C(=O)(C(C)S(C)(=O)=O)NCCN1CCN(C(c2c(OCC#C)nccc2)=O)CC1 22241,c1(C(=O)NCCCC2N(C(CC3CC(C)OC3C)=O)CCC2)c(F)ccnc1Cl 22242,C1(S(N)(=O)=O)(C(=O)NCC(C)N(C)C(c2cc(Cl)cn2C)=O)CCC1 22243,c1(C(=O)NCC2CC(F)CN2C(C2CCCC23CC3)=O)cnn2cnnc2c1 22244,Cc1nc(CCNC(c2cccnc2-n2nccn2)=O)c(C)o1 22245,c1(CCC)c(C(N2CCN(CCOCCC(C)C)CC2)=O)nnn1CC 22246,C1(N(C)C(C2CCOC2)=O)CCCN(C(c2cc(O)ccc2Br)=O)CC1 22247,C(=O)(C(O)CCC(F)(F)F)N1C(CN(C(=O)Cc2ncc(C)s2)CC)CCC1 22248,C1(NC(CC2C(C)(C)C2)=O)CC(NC(=O)OC(C)(C)C)C12CCC2 22249,N(C1CCC(NC(C2(n3ccnn3)CC2)=O)c2ccccc21)C(C(CCC)C)=O 22250,CC(C)C(CC(=O)NC1CCC(C2CC2)C1)NC(=O)CC1C(C)(C)C1(C)C 22251,C1(NC(CC(CCC)O)=O)CCCCN(C(c2cccc3cnsc23)=O)CC1 22252,c1(-c2nn(C(C)C3CC3)c(C(OC(F)(F)F)F)n2)ccc(F)c(Cl)c1 22253,C1(CCNC(Cn2ccc(C)n2)=O)CCN(C(C2CC2C(C)(F)F)=O)CC1 22254,C1(C(=O)NCc2ccon2)CC2CCCC2N1C(C1CC12CCCC2)=O 22255,N1(C(c2cc(CCC)on2)=O)CC2CCN(C(c3cncc(O)c3)=O)CC(C2)C1 22256,C1(NC(CCC(N)=O)=O)CC2(CCN(C(c3cncc(OC(F)F)c3)=O)CC2)C1 22257,c1(CC(=O)NCC(C)CNC(=O)Cn2cnc(C#N)n2)cc(F)ccc1F 22258,c1(NC(C2(c3ccccc3)CCC2)=O)cncn1C(F)(F)F 22259,N1(CC(=O)NCC2CCC2NC(C2C3CNC(=O)C23)=O)CCN(C2CC2)C1=O 22260,N1(C(COCCCC)=O)CC(CCNC(C2(C(C)C)CCC2)=O)OC(C)C1 22261,C1(c2scc(COC)n2)CCN(c2ccnc(NCCCC3CCOC3)n2)CC1 22262,N1(C(CCN(C(C)=O)C)=O)CCC(C)(CNC(=O)Cc2ccn(C)c2)C1 22263,c1(OC)cccc(F)c1C(=O)NCC1CN(C(=O)Cc2csc(C)n2)CCC1C 22264,C(=O)(C(O)CC(F)(F)F)NCC1N(C(CSc2nc(C)[nH]n2)=O)CCCC1 22265,C1(CCCNC(c2c(CC)noc2)=O)CCCCN1C(=O)C=CC1CCOCC1 22266,n1(CC)nnc(C(=O)NC2CC(CNC(c3cc[nH]c3)=O)C2(C)C)c1C 22267,C1(c2ccccc2)(NC(CC=C)=O)CCNCC1.C1(C=O)CCCS(=O)(=O)C1 22268,Cc1c(C(N2CCOC(C(=O)NCCC3OCCC3C)C2)=O)cnn1C 22269,C1(NC(C(C)C2CCCC2)=O)CCCCCN(C(c2cn3ccnc3cn2)=O)C1 22270,c1(OC)ccc(C=CC(=O)NC2CCCC2CNC(C2(O)CCC2)=O)c(OC)c1 22271,Cc1cc(NC(=O)NC2CC2(F)F)cc(F)c1Br 22272,Clc1cc2c(cc1Br)CCN(c1nc3c(Br)csc3s1)C2 22273,c1(N(C(=O)CNC(N2Cc3ncnc(O)c3C2)=O)C)cccc2ccccc12 22274,c1(C(N2C(CNC(CCN(CCC(C)(C)C)C)=O)CC2)=O)ccnc(Br)c1 22275,N1(C(C2C(=C)CC2)=O)CC(CNC(c2ncccc2C(=O)OC)=O)C(O)C1 22276,C1(CNC(C=CC)=O)(NC(=O)CSCC(N)=O)Cc2ccccc2C1 22277,C12(CNC(CCOCCC)=O)CC1CN(C(=O)C(C)Oc1ccccc1OC)C2 22278,Nc1cc(C(=O)NCC(c2cccc(Cl)c2)NC(c2csnc2Cl)=O)cc(F)c1 22279,N1(C(C2(COC)N(C(C(COC)OC)=O)CC=C2)=O)CCN(C)C(C)C1 22280,CCC(CCC(=O)N(C(C)CC(N)=O)C)NC(C1(C)CCCCC1)=O 22281,C#Cc1cccc(C(=O)NCC2COC(CNC(=O)C(C)(C)c3ccsc3)C2)c1 22282,C1(C(=O)NC(C(N2CCC(O)(CC(N)=O)C2)=O)CCOCCO)CCC(N=[N+]=[N-])C1 22283,CCCCC1CNC(=O)C=C2CCN(CC2)C(=O)CNC(=O)N1.C1(NC)CC1 22284,c1(OC)cc(C(N2CCN(C(C3CCCCN3C(C)=O)=O)CC2C)=O)cnc1C 22285,c1(CNC(C2CC(NC(CCNC(C)=O)=O)C2)=O)n[nH]cc1C 22286,N1(C(COCC)=O)CCC(C(F)F)(CNC(=O)C(C)Cc2ccncc2)C1 22287,c1(-c2c(F)cc(C)cc2F)ccc2c(C(=O)NCC(C)(C)C(N)=O)nn(C)c2c1 22288,c1(C(N(C(CNC(c2ccc(C(OC)OC)o2)=O)C)C)=O)occ2c1CCOC2 22289,CON1CCC(NC(C2(NC(=O)COCC3CCOC3)CC2(C)C)=O)CC1 22290,c1(CNC(=O)NCC2(COC)CCN(C)CC2)cn2cccc(Br)c2n1 22291,c1(C(N2C(CNC(C(C)O)=O)CCCC2)=O)cnc(C2CC2)[nH]c1=N 22292,Cc1cc(CCNC(=O)C(=O)NC2CC(CN)C2(C)C)c(C)s1 22293,CC(Cn1ccnc1)C(=O)NCC(O)C1(Cl)CC1 22294,C(=O)(CS(=O)(=O)C(C)C)N1CCC(N(C(=O)CCn2ccnc2C)CC#C)CC1 22295,c1(NCCS(CC)=O)[nH]c(=NC2CCc3oc(COC)cc3C2)nc2sccc12 22296,N1(C(c2ccn(C3CC3)n2)C(=O)NCC)CCc2c(cc(C#N)n2C)C1 22297,C1(CC(=O)NCC(C)(CO)NC(=O)C=CC2CCCO2)CCCCCCC1 22298,CC(c1ccc(F)cc1)=CC(N1CC(NC(c2c[nH]nc2[N+](=O)[O-])=O)C(C)C1)=O 22299,N1(C(COC(C)=O)=O)CCCC2CN(C(c3cc([N+](=O)[O-])oc3C)=O)CCC12 22300,C(=O)(C1=CC2CC=CCC12)N(CC(CNC(Cc1nc(C)sc1C)=O)(C)C)C 22301,C1(C(N(C)CCOCCN(C(=O)C(F)(F)c2cscn2)C)=O)CCCC(F)C1 22302,CC1CC(C2CN(C(C3CCC3NC(c3ccnnc3)=O)=O)C2)=NO1 22303,C1(n2ccc(C)n2)CCC(N=c2cc[nH]cc2S(=O)(=O)NCC=CCl)C1 22304,N1(C(c2c(C)nn(C)c2)=O)CCC2CN(S(=O)(=O)c3ccccc3F)CC2CC1 22305,CC1(c2cccc(CNC(=O)NCc3ncccn3)c2)NC(=O)NC1=O 22306,c1(OC)nc(Cl)ccc1C(=O)NCC1CN(C(c2cc3sccc3s2)=O)CC1O 22307,c1(OC)c[nH]nc1C(=O)NC(CN(C(=O)CC1C=CCC1)C)Cc1ccccc1 22308,N1(C(C(C2CCCCC2)NC(c2cn(C)c(=O)cc2)=O)=O)CC2(C)CC1CCO2 22309,Cc1cnccc1C(C)C(N1CC(NC(=O)CCc2cncnc2)CC1C)=O 22310,CC1(F)CN(C(c2csc3nccn23)=O)CCN(c2nc3cc(Cl)ccc3s2)C1 22311,N1(C(C(C)C2CCCO2)=O)C(CNC(c2n[nH]cc2Cl)=O)CC2COCC12 22312,c1(C(=O)NC2CCC3CCC23)n[nH]c2c1CN(C(c1cnc(Cl)s1)=O)C2 22313,N1(C(CN(C(C)C)C)=O)CCC2(CC2NC(=O)COC2CCCCCC2)C1 22314,CC1(C)CC(O)CCN(C(c2cc(F)cs2)C(=O)NC2CCOCC2)C1 22315,c1(C(C(=O)NCCN(C(=O)C=C(C)C(F)F)C)NC(COC)=O)ccccc1 22316,c1(NC(C)=O)ccc(C(=O)NC2COCC2NC(=O)CCc2nncs2)cc1 22317,N1(C(C(N2CCOCC2)C)=O)CCC(NC(=O)C2=C(Cl)CCC2)C1(C)C 22318,N1(C(C(C)N(C(=O)CC2OCCO2)C2CC2)=O)CC(CO)C(O)C1 22319,C1(CC)CN(C(=O)Cn2ccsc2=N)CCC1NC(c1ccnc(O)c1)=O 22320,n1(C(C)C)cc(Br)cc1C(=O)NC(C)CCNC(C1(O)CCSC1)=O 22321,Cc1c(C(N2CC3CN(C(=O)CCC(C)(C)C)C3C2)=O)cccc1O 22322,c1(C(=O)NC2C(C)CN(C(=O)C(F)(F)CC3CCCO3)C2)c(N)cccc1Cl 22323,CCCCC(C(=O)NCC1CC(C)=NO1)NC(=O)Cc1cnns1 22324,C1(C(=O)NC(C)CN(C)C(c2ccccc2)c2ccccc2)(OC)CC(C)(C)C1 22325,CCC(C)CC(C)C(=O)N(C)CCN(C(c1nn(C(F)F)cc1Cl)=O)C(C)C 22326,N1(C(Cc2cccc(OC)n2)=O)CCC(C)(C)C(NC(c2cccnc2S)=O)C1 22327,c1(C(C(=O)NCCC2N(C(C3COC(C)(C)O3)=O)CCC2)O)ccc(Cl)cc1F 22328,Cc1ccc(C)c(CNC(C2CC(O)(CNC(=O)C(O)Cc3cnc[nH]3)C2)=O)n1 22329,CC(C(C)C(=O)N1CCOCC1C(C)O)NC(=O)C(C)CC1CCCC1 22330,Cc1cc(C(=O)N(C)CCNC(c2cn(C)nc2C(F)F)=O)[nH]c1C 22331,c1(CC(N2CCOCC(C(=O)O)C2)=O)nc2c([nH]1)CCCC2 22332,Cc1cc(NC(=O)C(C2CCOCC2)O)ccc1NC(=O)C(C1CC1)N(C)C 22333,C1(C(=O)NCC(C)(C)OCCNC(C(C)Cn2ccnc2)=O)NC(=O)OC1C 22334,N1(C(Cn2cc(C(C)O)nn2)=O)CC(NC(c2cccn2C)=O)C2CCCCC12 22335,C=CCC(CNC(=O)C(C)OCC1CC1)C(=O)NC1(CO)CC2CCCC12 22336,N1(C(C2CCN(CC)CC2)=O)CCC2(CC1)CC(N1CCC(F)(F)CC1)C2 22337,c1(C(C)=O)cc(C(=O)NC2CC(C)(NC(c3sc(C4CC4)nc3C)=O)C2)c(C)o1 22338,C(C(F)(F)CNC(=O)CCCNC(=O)CC1(C)CC1)OC 22339,c1(C(=O)NCCC(C)NC(=O)C(=Cc2c[nH]cn2)F)cc2scc(Cl)c2[nH]1 22340,CC(C)C(C)C(CNC(c1cccc(C2(F)COC2)c1)=O)NC(=O)C1=COCC1 22341,OC1(F)CCN(C(=NCC2(O)CCCOC2)NCC2CCCCO2)CC1 22342,C1(OC)CN(C(C2(CCF)CCC2)=O)CC1NC(=O)CSC1CCOC1=O 22343,c1(OC)cc(C)c(C(=O)NC(CNC(=O)Cc2cnccc2C)C2CC2)c(C)c1 22344,Cc1nn(C)c(CS(=O)(=O)N(C(c2ccccc2)CCOC(F)(F)F)C)c1Br 22345,Cc1cc(CC(=O)NCC(C)(CO)NC(=O)CNC(=O)CCCCl)n[nH]1 22346,N1(C(C=C(C)C)=O)Cc2occ(C(N3CCC3CC3CC3)=O)c2C1 22347,c1(N2CC(C)(NC(C(C(C)O)C)=O)C2)nc2cc(Cl)cc(Cl)c2o1 22348,CC(C)(CO)C(=O)N1CCC(CCC(N2CCC(O)C2)=O)C1 22349,N1(C(c2sccc2Br)=O)CCN(c2ccc(-c3ccsc3C(F)(F)F)cc2)CC1 22350,CC1CN(C(c2ccc(OCC(N)=O)cc2)=O)CC1NC(=O)CCC1CC1(Cl)Cl 22351,Cc1nn(CC2CCC2)c(C)c1CC(=O)NN(C)CC1CCCN1C(C)C 22352,c1(NC(c2c(Cl)ccc(OC)c2)=O)ccc(S(C)(=O)=O)cc1Cl 22353,n1(CC(=O)NCC2CC2NC(C2CC2c2cccc(Cl)c2)=O)cccnc1=O 22354,C12(C(=O)NCC(CCC)NC(C3C4CN(C)CC34)=O)CC(C#N)(C1)C2 22355,c1(C(=O)NCCCCC=CCNC(c2nnn(C)n2)=O)ccc(O)c(Cl)n1 22356,C(=O)(C(C(C)C)C(C)C)N(C)CC1(C)C(NC(C(C(CC)O)C)=O)CCC1 22357,N1(C(c2c(SCC)cncc2)=O)CC2CC(NC(c3c(C)nn(C)c3C)=O)C2C1 22358,c1(C(=O)NCCC(C)NC(C(OC)OC)=O)ccc2cccnn12 22359,C1(C(=O)NC2(CO)CCCN(C(=O)CCCC3CC3)C2)(OC)CCS(=O)(=O)C1 22360,N1(C(CCCC(C)O)=O)CC(NC(c2csc(C3CCCO3)n2)=O)CC2(CC2)C1 22361,N1(C(c2cn(CC)nc2C)=O)CC(NC(=O)Cc2ccns2)C(N=[N+]=[N-])C1 22362,Cc1ncnc(N2CC3CC3(CNC(c3cc(F)ccc3Cl)=O)C2)c1Br 22363,C(c1cnc(C)s1)=CC(=O)NCC1(CNC(C(C=CCCC)O)=O)CC1(F)F 22364,CC(=Cn1ccnn1)C(=O)N1CC(C2CN(C(c3ccon3)=O)C2)C1 22365,c1(NC(c2ccsc2)CC)ccc(S(=O)(=O)NC2(C)CC2)cc1Br 22366,Cc1nn(C)c(C)c1NC(c1nc(Nc2nccc(C#N)n2)cn1C)=O 22367,C1(NC(c2ncn(CC)c2)=O)CCCC(NC(=O)Cn2nnc(C3CC3)n2)CC1 22368,N1(C(C(CCC=C)(F)F)=O)CCC2C(CCCN2C(=O)CC(F)(F)C(C)C)C1 22369,C12(O)CCN(CC1)C2=O.N1(CCNC(C2(C(=O)OC)CC2)=O)CC2CC2C1 22370,CC1OCCC1CNC(=O)C(C1CCCC1)NC(c1cscc1Cl)=O 22371,c1(C(=O)NC2C(OC)CN(C(c3cn(C4CC4)nn3)=O)C2)ccc(F)cc1O 22372,N1(C(C=C(C)Cl)=O)CC2C(NC(=O)CCSc3ccccn3)C2C1 22373,C=CC(C)(C)CC(=O)NC1CCCN(C(=O)CC2CCC(C3CC3)O2)C1 22374,Cc1c(C(N2CC3CC2C3C(=O)NCC2(O)CCN(C)C2)=O)cccc1F 22375,N1(C(c2c(C)nc(C(C)C)s2)=O)CC(NC(c2ccnc(CO)c2)=O)C2CC2C1 22376,C=CCC(CC(=O)NC(CCC)c1nn[nH]n1)NC(=O)CCCF 22377,C(=O)(CS(=O)(=O)N(C)C)NCCOCCN(C(=O)C(F)(F)c1cncs1)C 22378,N1(C(C2CC(C#C)(O)C2)=O)CCC(O)C(NC(c2cnsn2)=O)C1 22379,c1(C(=O)NCC2CC(NC(c3cccnn3)=O)C2)cnc(S)nc1 22380,C12(CNC(COCC#C)=O)CCC(CC1)N2C(C1(C)CNC(=O)C1)=O 22381,n1(CCCC)c(C)cc(C=C(C#N)C(=O)Nc2c(C(N)=O)noc2C)c1C 22382,N1(C(=O)C=CC=Cc2ccccc2)CCC(CNC(C2COC(=O)C2)=O)C(O)C1 22383,c1(C(N(CCNC(=O)Cc2ccsc2Cl)CCOCCO)=O)ccc2c[nH]nc2c1 22384,N1(CCN2C(CF)CC(OC)C2)CC2C(c3ccccc3)(C1)CS2(=O)=O 22385,CCCCCCC(F)C(=O)NC1CCC12CCN(C(=O)CCSCC(N)=O)CC2 22386,N1(C(C(C)n2ccnc2)=O)CCCN(C(=O)C2=CCCS2)C(c2ccccc2)C1 22387,c1(-n2cc(CC(=O)NC(c3cnc(C)s3)C(=O)O)nn2)ccc2c(c1)OCCO2 22388,C1(C(N(C2CC(O)C2)C)=O)C=CCN(C(=O)CC2OCCCO2)C1 22389,C(=O)(C(C(C)(C)O)NC(c1cccn(C)c1=O)=O)NC(C(=O)OC)CO 22390,c1(N2CCCC3(CC(NC(=O)C4CCCc5n[nH]cc54)C3)C2)nc2ncc(Cl)cc2s1 22391,N#Cc1cc(F)ccc1C(N1CCN(C(C2CCSCC2)=O)C2CC12)=O 22392,Cc1ccc(CC(N2CCCC(O)(CNC(=O)C(C(C)O)N(C)C)C2)=O)cc1C 22393,N1(C(c2c(C)ccnn2)=O)CCN(C(=O)C(C)(F)C(C)(C)F)CC12CCC2 22394,C(=O)(CCC(CC)OC)NC(CC#C)C(=O)NCCC1CCOCC1 22395,n1(CC)cc(CC(=O)NC(C(=O)NC(C)CC2CCC2)C2CCOC2)cn1 22396,CC(C1CCCCC1)=CC(=O)NC1CN(C(=O)COC2CC=CC2)CCC1C 22397,c1(C(=O)NC2CC(F)(CNC(C(n3ccc(C)n3)(C)C)=O)C2)cccn(C)c1=O 22398,C(=O)(C(C(=O)NC1CC2(C(=O)NC3CCOCC3C)COC1C2)C(C)C)OCC 22399,n1(CC(=O)NC2CCC(NC(C(CC)O)=O)C2)nc(-c2ccccc2)oc1=O 22400,c1(CC(=O)NC)ccc(C(=O)NC2(C)CN(C(=O)CC(C)(C)O)C2)cc1 22401,c1(CNC2CC(C(=O)NC3(CCC)CCNC3=O)OCC2)ccc2n[nH]cc2c1 22402,N1(C(C(CC#C)(C)NC(=O)CCC#CC)=O)CC2(CNC(=O)C2)C1 22403,N1(C(C=C(C)C(C)C)=O)CCC(O)(C(C)NC(=O)CCOC(C)CC(C)C)CC1 22404,C1(C(=O)NC(CC)C(C)(F)F)CN(C(=O)C(C)O)CC1C1CC1 22405,c1(C(=O)NC2(C)CC(NC(=O)CC3COC4CC3C4)C2)cc([N+](=O)[O-])ccc1Cl 22406,C(C(C)(C)C(=O)NCCC(C)CCNC(=O)C=C1CCCC1)OCC 22407,CC1(C)CN(C(=O)CC2CC3(CCC3)C2)CC(CNC(=O)COCC2CC2)O1 22408,Cc1ncc(Cl)c(C(N2CC3C(CNC(=O)C(C)(C)O)C3C2)=O)n1 22409,N1(C(C2(F)CCN(C(C(CC=C)N(C(C)=O)CC)=O)CC2)=O)CC(C)N(C)CC1C 22410,c1(C(N2CC(C(=O)NCCc3ccc(OC)nc3)C(C)C2)=O)cccc(C#N)c1 22411,c12cc(c(C)o1)S(=O)(=O)NC2=O.N1(CCC)C(=O)CCC1C(=O)NC 22412,C(=O)(C1=NN2CCCN=C2N1)NCC1CN(C(CSC(C)C)=O)CC1(C)C 22413,C1(CNC(c2nnc(C(F)(F)F)s2)=O)C(O)C(O)CN1C(=O)CCC(F)(F)F 22414,c1(CC)nn(C)c(NC(C2C3CN(C(=O)CCS(=O)(=O)N(C)C)CC23)=O)c1Cl 22415,c1(C(=O)NC2C3CN(C(C4(CF)CC4(F)F)=O)CC23)cccc2cnccc12 22416,C1(C2CCCC2)(C(N2CCN(C(C(C)SC)=O)CC2)=O)CCNC1=O 22417,C1(NC(c2cnc3cccnn23)=O)CCc2nnc(C(F)(F)F)n2C1 22418,N1(C(CNC(C(C)(C)C)=O)=O)CCC2CCCC12C(N1CCCC(C)(CO)C1)=O 22419,Cc1nsc(C(=O)NC2(CF)CN(C(=O)CCc3ccccc3)C2)c1N 22420,C1(CCCNC(=O)CSc2cccnc2)CCCCN1C(c1cccnc1)=O 22421,c1(CC(N2CCC(N(C(CC(CC)OC)=O)C)C2)=O)c(F)cccc1Cl 22422,C1(CC(=O)NCC(C23CCC(CC2)C3)NC(c2ccoc2)=O)CCCNC1=O 22423,CC1CN(C(C2(c3ccccc3Br)CCC2)=O)CCN1C(C1C=CCCC1)=O 22424,C1(C)(C(=O)NCC(C)(C2CCC2)NC(Cn2ncc(C)c2)=O)COCCO1 22425,C(CNC(=O)CC1(O)CCC1)(CC(=O)N1CCC1(C)C(=O)OC)OC 22426,N1(C(C(CC)OC)=O)CCOC(C(=O)NCC2(F)CC(CO)C2)CC1 22427,CCC(C(=O)OC)C(=O)NC1CC=C(C(=O)NCCc2nc(C)no2)C1 22428,c1(NC(=O)CCSC2CCCC2)ncnc2[nH]cc(Cl)c12 22429,Cc1ccc2c(C(=O)NCC3CC3NC(c3cc(N(C)C)ccn3)=O)n[nH]c2c1 22430,C1(COC)(CNC(=O)CC#N)CCN(C(=O)Cc2ncccc2C)C1 22431,c1(C(=O)NCCC2(O)CN(C(C34CCCC3CC4)=O)C2)cnc2n1CCOC2 22432,S(=O)(=O)(CCN=c1ccnc(NCC(c2nc(C)cs2)(C)C)[nH]1)NCC 22433,N1(C(C(C)C)=O)CCCC(NC(=O)CC(c2ccc(C(F)(F)F)cc2)C)C1 22434,C(=O)(C1=C2CCCN=C2NN1)N1C2C(NC(c3n[nH]c(C)c3C)=O)CC(CC2)C1 22435,c1(OCOC)cccc(C(=O)NC(C)CNC(=O)C(F)C(C)C)c1 22436,Cn1cc(C(N2CCC(CNC(=O)Cc3cscn3)C2)=O)nc1C(F)F 22437,N1(C(C(C)OCCOC)=O)CCCC1C1(NC(=O)Cn2cc(C(C)=O)nn2)CC1 22438,c1(C(=O)NC(CN(C(C(C(CC)C)O)=O)C)CC)ccc2cccnc2c1 22439,C(=O)(C1=C(Cl)CCC(C)C1)N1CCC(NC(CN(C(=O)OCC)C)=O)CC1C 22440,C1(NC(CC2CN(C)C2)=O)CCCC(NC(=O)C=Cc2cccc(F)c2)CC1 22441,c1(C(C)(C)C)nc(=N)[nH]c(=NC2C3CC2CN(C(=O)C2=CCCCCC2)C3)[nH]1 22442,CC(C(=O)N1CCC(C(CO)NC(=O)C(C)(F)c2ccon2)CC1)S(N)(=O)=O 22443,N1(C(c2cn(CC)nn2)=O)CC2(CCC2NC(=O)CC2CC3(CC3)CO2)C1 22444,Cc1ccc(C2(C(N3CCC(NC(C4CC4C#N)=O)C3)=O)CCOCC2)cc1 22445,C(=O)(C(CC(F)F)c1ccccc1)NC(C(C)NC(c1n(CC)ncc1)=O)(C)C 22446,CC1=C(C(=O)N(CC(=O)NC2N(C)CCCC2(C)C)C(C)(C)C)C(=O)OC1(C)C 22447,CC1CC(NC(=O)C(C)(C)N2CCOCC2)CCN1C(C1C(F)(F)C12CC2)=O 22448,C1(NC(CCOCC)=O)CN(C(=O)C=CC2CCOC2)CC12CC2 22449,c1(CC)c(C(=O)NC(CNC(=O)CC(C)C(F)F)CO)cccc1C 22450,c1(C(N2CCC(N(C(C(C)OCC=C)=O)CCO)C2)=O)ccc2c(c1)CCC=C2 22451,C1(NC(C2N(CC)CCC2)=O)CN(C(c2cccc(=O)n2C)=O)C(C)(C)C1 22452,c1(CC)nnc(C)cc1C(N1CC(NC(c2cn(C)c(=O)n2C)=O)CC(C)C1)=O 22453,N1(CC)CCC(NC(C2CCOCC2NC(C2CC2Cl)=O)=O)C1=O 22454,C12(NC(COC(C)=O)=O)CCCC(NC(=O)Cc3nccn3C)(C1)C2 22455,C(=O)(C(CC)C(C)(C)CC)NC1C2(CCN(C(CCC=CCC=C)=O)CC2)C1 22456,C(=O)(C#CC(C)(C)C)NCC(C)(CO)NC(CC(C)c1ccncc1)=O 22457,N1(C(CSC)=O)CCC2(NC(=O)CC3CCCC3C)CCCC12 22458,N1(C(C2(C)CC(C)C2)=O)CCC(C2(O)CN(C(C3C4COCC34)=O)C2)CC1 22459,c1(CC)cc(F)ccc1CC(=O)N(CC(CC)NC(=O)Cc1ncoc1C)C 22460,C1(NC(=O)CCc2ccsc2)CCC2(CCCN2C(C2CCCS2)=O)CC1 22461,c1(CSc2nc3ccc(C(=O)OC)cc3o2)nc2ccc(Br)cc2n1C 22462,C1(F)(C(NOC(C(=O)NCc2ncc(COC)s2)C)=O)CCCCC1 22463,c1(C(=O)NCCCN(C(c2c(SC)scc2)=O)C(C)C)cn(C)nc1C(N)=O 22464,c1(OC)cccc(CC(C)(C)NCc2c[nH]nc2C(F)(F)F)c1 22465,n1(C(C)C)ccc(C(N2CCC2CNC(c2nc(Cl)cs2)=O)=O)n1 22466,N1(C(CCC#C)=O)CC(CCNC(c2ccnc(Cn3cnnc3)c2)=O)OC(C)C1 22467,C1(C(=O)NCC2C(C)CN(C(=O)C=CC3CC3)C2)C2CCCCCCC12 22468,N1(C(C(C)C#N)=O)CC(C2CCCN(C(C3CC(c4ccccn4)=NO3)=O)C2)C1 22469,Cc1[nH]ccc1C(=O)N(C1CC1)Cc1cn(CC(N2CCC2CN=[N+]=[N-])=O)nn1 22470,c1(C(N(CCCNC(CCOCCC)=O)C)=O)cc(Cl)c(C)cc1OC 22471,C1(OC)CCN(C(c2n[nH]cc2CNC(=O)C(C)OC2CCCC2)=O)C(C)C1 22472,c1(C(N2CC(NC(c3ccc(OC)o3)=O)C(CO)C2)=O)nccc(C)c1F 22473,Cc1cc(C)[nH]c(=NCC2(N(C)C(c3cccn4c(O)nnc34)=O)CC2)n1 22474,C1(CC(=O)NC(C(C)(C)NC(c2cncc(COC)c2)=O)C)NC(=O)CNC1=O 22475,CC(N=c1cc(C(F)(F)F)nc(Cl)[nH]1)C1CCCN(C(=O)C=Cc2nccs2)C1 22476,CCCCC(O)CC(=O)NCC1(Nc2cn(CCCF)nn2)CC(OC)C1 22477,n1(CC)cc(Cl)cc1C(=O)NC1(CNC(C23COCC(C2)C3)=O)CCCC1 22478,c1(C(N2CC3C(NC(c4c(OC)n[nH]c4)=O)C3C2)=O)cc(Br)cc2cc[nH]c12 22479,c1(C(N2CCOCC2)C(=O)OC2(C(=O)OCc3ccccc3)COC2)cc(Cl)cs1 22480,CCS(=O)(=O)c1cccnc1C(=O)NCC(C)(N)Cn1cc(Br)cn1 22481,C(C)(C(CC(=O)NOC(c1ccco1)CO)NC(c1ccco1)=O)OC.C1(=O)CO1 22482,N1(CCC)CCC(C(=O)NC2C3CC(NC(=O)Cc4ccsc4)CC23)CC1 22483,Cc1ccc2c(c1)C(C(=O)N(CCCN(C)C(C1CCCSC1)=O)C)C2 22484,N1(C(C2CC(C)(C)C2)=O)CC(CNC(=O)CC2=CCCCC2)C2(CCOCC2)C1 22485,c1(OCC)ccc(NC(C2=CCSC2)c2nnnn2CC2CCCO2)cc1CO 22486,N1(C(C(CC)(C)C)=O)CCC(NC(=O)Cc2cc(Cl)ccc2O)C(C)C1 22487,c1(C(=O)NCC(C)NC(c2c(C)nn(C3CC3)c2)=O)cnn2c(N)ccnc12 22488,C(=O)(C(=O)C(C)(C)C)N(C(C(=O)Nc1ccsc1)C1CC1c1cccc(I)c1)C 22489,N1(C(=O)CN2CCOCC2)CCCC(CCC(=O)NCC23CC(CO)(CO2)C3)C1 22490,c1(CCC(=O)NCC2(OC)CN(C(=O)C(C)CO)C2)ccc(C#N)cc1 22491,C(C(CC(C)C)C(=O)N(C(C)CN(C)C(c1cnc(Cl)n1C)=O)C)OC 22492,Cc1cc(N2CCC(C(C)NC(C3CCCC(O)C3)=O)C2)c(Br)cc1[N+](=O)[O-] 22493,c1(C(=O)NCC2(NC(=O)C3=CCSC3)CC2)c(Cl)ccc(Br)c1F 22494,C12(NC(CN(C)C)=O)CCCCCC1N(C(c1coc(Br)n1)=O)CC2 22495,Cc1cnn(C)c1CC(N1CC(C)(NC(=O)CCC=CBr)C1)=O 22496,C1(CN(C(C(C2CC2)OC)=O)C)CCCN(C(=O)CCCOC(C)(C)C)C1 22497,CC1(C)CC(NC(=O)C(C2CCOCC2)F)CN(C(=O)Cc2cc[nH]c2)C1 22498,c1(OC)cc(CN(CC(C)(C)C2(O)CNC2)C=O)cc(F)c1 22499,c1(-c2c(C)c(N3CCn4c(C)cnc4C3)ncn2)cccc2c1OCCO2 22500,CC(C)(O)C(F)C(=O)NCC1CCCCC1C(N1CC2(CCC2O)C1)=O 22501,Cc1cc2nc(NCC3CC4(CC(NC(=O)C(F)(F)Br)C4)C3)cc(=O)n2o1 22502,N1(C(c2cccc(OC)n2)=O)CCC(F)CC1C(=O)NCC1CC(C)(C)CCO1 22503,C1(NC(C(c2cccnc2)N(C(C)CCO)C)=O)CCCCC1N1CCOCC1 22504,N1(C(C2CC3(CC(NC(C(CC(C)(C)C)OC)=O)C3)C2)=O)CCC2(CCC(O)C2)C1 22505,C1(NC(C(c2ccc(F)cc2)C)=O)C2CC(CN(C(=O)C=C3CCC3)C2)C1CO 22506,N1(C(c2ccc(NC(C)=O)cn2)=O)CCCC(NC(=O)C(F)(F)CC2CC2)C1C 22507,C(=O)(C(C)CC(F)F)N1CC(CCNC(c2c(C)[nH]c(=N)s2)=O)C1 22508,C(=O)(C(C)CC(C)(F)F)NC(CCNC(CCc1ccc(OC)cc1)=O)C(C)C 22509,C(CCCC(C)C)NC(CCC1N(C(c2c(C)scn2)=O)CCC1)=O 22510,C1(C(N2CCC(OCCO)C2)=O)(CNC(C2N(C)CCC2)=O)CCCCC1 22511,c1(C(=O)NC(C)C(=O)Nc2cncc(-c3ccco3)c2)nc2ccccc2s1 22512,N1(C(c2c(C)cc(SC)o2)=O)CC(NC(=O)Cc2coc(C)n2)CC1(C)C 22513,C1(CC)(N)CNC1.C1(C(=O)C(c2cccnc2)=O)CCC(OC)C1 22514,c1(CNC(C(C2CCN(C(=O)CCNS(C)(=O)=O)CC2)C)=O)ccc(O)c(O)c1 22515,c1(CC(=O)NCCN(C(C=C(CC)C)=O)CCOC)cccc(C(C)OC)c1 22516,N=c1ncn(CC(=O)NC(CC2CCC2)C(=O)NC(CC2CCC2)CO)[nH]1 22517,C1(NC(C2(N(C)C)CCCC2)=O)CN(C(=O)CC2CCC23CCC3)CC1C(F)F 22518,c1(N2C(CC)C(C)(C)C2)ncnc2c1ncn2C(C1(O)CCOC1)C1CC1 22519,CCC(CC)(CC)C(=O)N1CC(C)(c2cn(-c3ccc(C(C)(C)C)cc3)nn2)C1 22520,CCC(CC)CC(=O)NCC12CC1CN(C(=O)CC1(C)CC1(F)F)C2 22521,C12(C(N3CCC(C)(NC(c4c(CC)noc4)=O)C3)=O)CCOC1CC(=O)NC2 22522,C(=O)(C(COC)OCc1ccccc1)NC(CNC(C=CC(CC)=CC)=O)C 22523,c1(N2CCCC(C(C)C)C2)nc(=NC2CCCc3n[nH]cc32)[nH]c2c1COCC2 22524,c1(C(C)C)ncncc1C(=O)NCC1CC(NC(=O)CC(C)C2CC2)C1 22525,N1(C(C2(OC)CC2)=O)CCOCC(NC(c2cc(Br)no2)=O)C1 22526,c1(C(N2CCC(CN(C(C(C(=C)C)(C)C)=O)C)C2)=O)ccc([N+](=O)[O-])c(C)n1 22527,C1(N(C(=O)C=CBr)C)CCCCN(C(=O)C(C)(C)c2ccno2)C1 22528,C1(CNC(C)=O)CCCN(C(C2(n3cc(CC(C)O)nn3)CC2)=O)C1 22529,c1(C(=O)NCC(C2CC2)NC(c2ccc(CC)[nH]2)=O)ccc(=O)n(CC(C)O)c1 22530,c1(CCC(=O)NCC2(C(=O)OC)CC2(F)F)cccc(F)c1Br 22531,C1(NC(C(=CC2CCCC2)C)=O)CN(C(=O)C(F)=CCCF)CCC12CCC2 22532,N1(C(Cc2c(C)n[nH]c2)=O)CC(CNC(=O)CCC2CCCO2)C(C)(C)C1 22533,C(=O)(CC(C)(C)C(=O)N1CC2C(CNC(C3CCS(=O)CC3)=O)C2C1)OCC 22534,O(NC(=O)C(CC(C)C)NC(C1CCCC(=O)N1C)=O)CC 22535,c1(NCC)ncc(C(=O)NC23CC(CNC(=O)C#CC(C)C)(C2)C3)cc1Cl 22536,c1(CC(=O)NCC23CC(NC(C(COC)N(C)C)=O)(C2)C3)c(O)ncnc1O 22537,c1(C(=O)NC2CN(C(CNC(=O)OCC)=O)CC(F)C2)csc2ccc(F)cc12 22538,CCCC(C)CC(=O)NC(C)C(C)NC(c1onc(OC)c1Br)=O 22539,c1(OCC)cccnc1C(=O)NCCC(C)N(C(=O)C=Cc1ccc[nH]1)C 22540,C1(C)(CNC(C(CC)O)=O)COCCN(C(c2cc(F)c(O)c(Cl)c2)=O)C1 22541,C(C(=O)N1CCCC1CC(=O)O)(C(C)C)N(C(=O)OC)C 22542,N1(C(CC2CC(C)C2)=O)CC2(CNC(c3cnn(C)c3Cl)=O)CC1CO2 22543,C=C(C)C(C)(C)C(=O)NCC1(C)CC(NC(=O)C(C(C)C)SC)C1 22544,c1(C(=O)NCC(CO)NC(C(C2CC2)OC)=O)c[nH]c(=N)nc1C 22545,c1(C(=O)NC2(C)CC(C(N3CCCN(C(C)=O)CC3)=O)C2)cc2ccccn2c1 22546,CC(C)CC(O)C(=O)NC1(C(=O)NC2CCCCCC2C)CC1(C)C 22547,CC(CC(C)(C)C)C(F)C(=O)NCC1C2CN(C(c3ccc(F)s3)=O)CC12 22548,N=c1[nH]c2ccc(C(=O)NC3CCCC3NC(c3ccccc3)=O)cc2[nH]1 22549,C=C(Cl)CN=c1ccc(S(=O)(=O)N(CC)CC2CCN(CC)CC2C)c[nH]1 22550,CCCCCC(O)C(=O)N1CC=CC1CNC(=O)CNC(C1CCC1)=O 22551,c1(CC(=O)NC2CCCC2Cn2cc(-c3ccns3)nn2)ccc(F)nc1F 22552,C(=O)(C1=CCCOC1)NCCC1CCC(NC(CC(CC)c2ccccc2)=O)C1 22553,c1(C(C)(C)C)cncc(NC(C2CN(C(=O)C3CC3)CCN2)=O)c1 22554,C1(C(=O)NCC=CCCC)N(C(=O)Cn2nnc(C)n2)CCCC1(C)C 22555,c1(C(N2CC(C(Cn3cc(CSC)nn3)F)C2)=O)ccc2nc(Cl)nn2c1 22556,c1(C(=O)NC2(CNC(C(CC)C(C)C)=O)CCCCCC2)ncnc2c1CCC2 22557,c1(-n2c(C(CC#C)C)nc(C(C)CCC)n2)ccc(S(=O)(=O)N(C)CC)cc1 22558,N1(C(CC(C)=C(C)C)=O)CC2CC(CNC(C3(n4cccc4)CC3)=O)C2C1 22559,N1(C(c2n[nH]c(C)c2O)=O)CCC(C2CC2)(CNC(=O)COc2ccccc2)C1 22560,C1(C(=O)NCC(CC)C)CC(C)CN(C(C2CCC(O)CN2C)=O)C1 22561,N1(C(CN(C(=O)COCC2CCCO2)CC#C)=O)CC2COC(=O)C2C1 22562,N1(C(C23C(CN(C(C(CC#C)OC)=O)C2)C3)=O)CCCSCC1C 22563,c1(C(N2CCC(O)(CCNC(CSCC=C)=O)C2)=O)cccc(C(N)=O)c1F 22564,c1(OCC)nc(N2CC(CNC(c3ccccc3SCC)=O)CC2C)ncc1C 22565,C1(C)(C(=O)NCC2CC(NC(c3c(C)cnn3C(C)C)=O)C2)CCCNS1(=O)=O 22566,N1(C(c2cnc(SC)s2)=O)CCC2CN(C(=O)CC(C)CF)C2C1 22567,C1(C(=O)Nc2cnc(I)cn2)CCN(Cc2ccc(OCCO)cc2)CC1O 22568,C(C(O)(C(F)(F)F)c1cccc(Cl)c1)NC(=O)NC(C(C)F)C(=O)O 22569,N1(C(c2c(CCC)n[nH]c2)=O)CC=CC(NC(c2cnco2)=O)C1 22570,Cc1cc(C)n2ncc(C(=O)N(C(=O)C(N3CC4CCC(N)CC4C3)=O)CC)c2n1 22571,C(=O)(CS(=O)(=O)CC1CCCO1)NCC(C(C)(C)C)NC(=O)C=C1CCCC1 22572,c1(NC(=O)NCC2(C=C)CCOCC2)cncc2sccc12 22573,C(CCC)(C(=O)NCC(C)CNC(C1(CC(C)C)CCCC1)=O)=CCC 22574,c1(-n2cc(NCC3CCCN(C(C(COCC)O)=O)C3)nn2)ccc(C)c(Cl)c1 22575,Cc1cc(C)n(CC(N2CCC(N(C)C(c3cccc(CS(C)=O)c3)=O)C2)=O)n1 22576,C1(C(=O)NC(C(=O)OC)C)CN(C(c2ccc(COC(C)=O)s2)=O)CCC1O 22577,N1(C(C(F)=CCC)=O)CC(C)N(C(c2ccc(C3OCCO3)cc2)=O)CC1C 22578,O=C(N=c1ccn(C(F)F)[nH]1)C1COC2(C1)CN(C(c1ccc(Cl)nc1I)=O)C2 22579,N1(C(CC=CC)=O)CCC(C)(CC(=O)N(C(C2CCC2)C)CC)C1 22580,N1(C(c2ccn(CCNC(C3(CC)CCC3)=O)c2)=O)CC(S(N)(=O)=O)C1 22581,CC1(C(=O)NC2CCOC(CNC(=O)CCc3cccnc3Cl)C2)COCCO1 22582,N1(C(c2nn(CC)c(O)c2)=O)CC2CCCC2(CNC(=O)C2=NOC(C)C2)C1 22583,c1(NC(=O)NC(c2ccccn2)Cc2cccc(C)c2)cc(F)c(I)c(F)c1 22584,N1(C(C(C)(C)CC(F)F)=O)CC(NC(=O)CCc2cnco2)CC2(CCC2)C1 22585,C(CN=c1[nH]cc2ncnc-2[nH]1)=CCNC(c1cc2ccncc2s1)=O 22586,C1(NC(C(CC)N(C)C)=O)CCN(C(C2CC(=O)NC2(C)C)=O)C12CCC2 22587,C1(N(C)C(C2C=CCS2)=O)CN(C(c2cc(Cl)c[nH]2)=O)CCC1O 22588,C1(N(C(=O)C(O)C2CN(C(C3CCCC3F)=O)C2)CC)CCCCC1 22589,CC(C)CCCC(C)CCNC(=O)N(C(C)C(C)O)Cc1ccc(Cl)cc1 22590,c1(C(=O)NCCC2(O)CCN(C(=O)CSC(F)F)C2)cnn2ncccc12 22591,C(=O)(C(C)(O)COC)NC1CC(C)(NC(c2ccc(CC)cc2)=O)C1 22592,c1(C(C(=O)NCC)N(C2CCC2C)C)cc2c(cc1OC)CCC2 22593,C1(C(N(CC(O)C2CCC2)C)=O)CCC(NC(=O)C(C2(O)CCCC2)F)C1 22594,Cc1cc(NC(=O)C(C)CNC(=O)Cc2cnccc2C)c(C)c(C)c1 22595,N1(C(C2(C)CCCOC2)=O)CCOC2(CCN(C(C3CCC4CC4C3)=O)C2)C1 22596,C1(C(=O)NCC=C2CCSCC2)(NC(C(c2cncnc2)C)=O)CC(O)C1 22597,O=C(CC(F)(F)F)NCC1CC(NC(=O)CCCOc2cccnc2)C1 22598,c1(C(N2C(C(=O)Nc3nnc(C)o3)CC2)=O)c(C)[nH]c2ccccc12 22599,c1(C(N(C2CN(C(C34CC(C3)C4)=O)C2)C)=O)cc(O)c(O)c(O)c1 22600,C1(C(N2CC(NC(CN(C(C)=O)C)=O)(CO)C2)=O)CCC(=O)N1C 22601,c1(C(=O)NC2(CNC(=O)Cc3csc(-c4cccs4)n3)CC2)ncc[nH]c1=O 22602,C1(NC(c2nccc(CC)c2)=O)CC2CC1N(C(c1ccc(F)c(N)c1)=O)C2 22603,c1(C(=O)OC(c2nccn2C)C)ccc(=O)n(CCN(C)C)c1 22604,C=CCC(CNC(=O)CC1(C#N)CC1)C(=O)NC(C)Cc1nncn1C 22605,C(=O)(C1=CC2(CCOCC2)C1)NCC(C)CNC(=O)C(CO)C(C)(C)C 22606,C(C(C)(C(=O)N(CC(O)CNC(c1n[nH]cc1I)=O)C)OC)OC 22607,N1(C(C(C2CCC2)NC(c2c(OC)ccnc2)=O)=O)CCC(C)C(F)(F)C1 22608,N1(S(=O)(=O)c2cnccc2N2C3CCC2CC3)Cc2ccccc2CC1CO 22609,N1(C(C(CC)(C)O)=O)C2CCC1CN(C(c1cc(O)ccc1Br)=O)C2 22610,C1(C)(C(=O)NCC2(F)CC(NC(CSCCOC)=O)C2)CCC(=O)N(C)C1 22611,CN1CCCC1(C)C(=O)NCC(c1cccc(Cl)c1)NC(C1(C2CC2)CC1)=O 22612,N1(C(c2ncc(NC)nc2)=O)CC(C)C(C)(CNC(=O)COC(C)C)C1 22613,Cc1ccc(NC(C2C=CC(NC(=O)Cc3c(F)cccc3F)C2)=O)c(CO)n1 22614,Cc1cc(C(N2CCCCC2CNC(=O)CNC(=O)C(C)C)=O)cc(C(F)F)c1 22615,Cc1oc([N+](=O)[O-])cc1C(=O)NCCC(C)(C)NC(=O)C(=Cc1cscn1)F 22616,C(=O)(C1=C(C)S(=O)(=O)CC1)NC1CN(C(c2c(C#C)c[nH]n2)=O)C(C)(CC)C1 22617,C1(C)(CC(=O)N(CCC(C)NC(COCC(C)C)=O)C)CCCC1 22618,c12ccc(O)c(c1)S2.C12(COCC)OCC(CNC=O)(C1)C2.C1(C)C(=O)N1 22619,N1(C(c2cnnc(C)c2C)=O)CCOC2CN(C(C3CCN(C)C(=O)C3)=O)CC12 22620,c1(NC(C2N(C(c3c(C)nn[nH]3)=O)CC(O)C2)=O)ncc(Br)cc1F 22621,Cc1cc(C(N2CCN(C)CC2CNC(c2c(Cl)nsc2Cl)=O)=O)cc(=O)n1C 22622,c1(C(=O)NC2CC(NC(CCCOC)=O)C2)cc(C)c(Br)cc1C 22623,N1(C(c2nccc(C)c2)=O)CCN(Cc2ncccc2C(F)(F)F)CC1C#N 22624,C#CCC(C(=O)NCC1(NC(=O)C=CC2CCCCC2)CCOC1)C1CC1 22625,C1(NC(C2CC(C)CC(C)(C)C2)=O)CCC2(CC1)CN(C(=O)CSS(C)(=O)=O)C2 22626,CCC(CC)(CC)C(=O)NC1CN(C(=O)CS(=O)(=O)CC)CC1O 22627,C1(S(C)(=O)=O)(C(=O)NC2CC(NC(c3nc(N(C)C)nc(O)c3)=O)C2)CC(O)C1 22628,C#CC1CCN(C(=O)C(Cc2cn[nH]c2)NC(=O)CCCN(C)C(C)=O)C1 22629,Cc1cn2c(C)c(C(=O)NC(C)(C)CN(C(=O)CCCN(C)C(C)=O)C)nc2s1 22630,C1(C(=O)NCCNC(N)=O)CCC(O)CN1C(=O)Cc1cccc(O)c1 22631,S(=O)(=O)(c1ccccc1Br)N1CCC(C(N2CCCC(C#C)CC2)=O)CC1 22632,c1(OC(C)C(=O)N2CC(CC(=O)NC3CC4CC4C3)C2)ccccc1 22633,CC1COC2(C1)CN(C(=O)C(C1(C)CC1)NC(C1CN(C)CCO1)=O)C2 22634,C1(C2CC2)(CNC(CCSCC)=O)CCN(C(c2cn(C)nc2Cl)=O)C1 22635,N1(C(C(C(CC)O)C)=O)CCc2nc[nH]c2C12CCN(C(c1csc(C)n1)=O)C2 22636,C1(C(=O)NC2C(COCC(=O)NCC(=O)NC3CC3)C2)CCCO1 22637,Cc1nc(N(C2CC3CNCC3C2)C(c2ccccc2C2CC2)=O)cc(C2CC2)n1 22638,C1(O)(C(C(=O)NCC(C#C)OC)NC(=O)C(C)(C)OC)CCCCC1 22639,C1(NC(c2cc(Cl)nnc2O)=O)CN(C(=O)CSCC(F)(F)F)CC1C1CC1 22640,CC(C)(CC(=O)NCC1CCCCN(C(C2CCC(N=[N+]=[N-])C2)=O)C1)CC(F)F 22641,C1(F)(C(=O)NCC2N(C(C)=O)CCC2)CCN(C(C2(C)CCN(C)C2)=O)C1 22642,N1(C(C2(CCC)CC2)=O)CCC(F)(F)C(CNC(C2(SC)CC2)=O)C1 22643,CC1=CC(C)CN(c2cc(C)nc(NC(C3CCOC3)COC(C)(C)C)n2)C1 22644,c1(C(=O)NCC(CNC(Cn2ccc(C)cc2=O)=O)(C)C)cncc2nc[nH]c12 22645,C(CC(C(=O)NC1(CCCCNC(c2csc(Cl)c2)=O)CC1)OC)OC 22646,C1(CNC(c2cc(Br)ccn2)=O)CCCCN(C(C2CC3(CCCC3)C2)=O)C1 22647,c1(C(N(C)CC2N(C(C(C=C)C)=O)CCCC2)=O)cc(CC)ccc1F 22648,CCC(C)(C)CCCC(=O)NC(CC)CCCC(=O)NC1(C2CC2)CC1 22649,c1(C(N(C2CCN(Cc3cc(OC)ns3)C2)C)=O)cc(F)c2ncccc2c1 22650,C1(CC)C(C(=O)NCc2nc[nH]n2)CCN1C(C1CC(F)(F)C1)=O 22651,C1(CN(C(=O)Cn2ncccc2=O)C)CCN(C(C2(N(C)C)CC(O)C2)=O)CC1 22652,C(C(C)C(C)(C)C)N(C(C)C)C(C1CCCN(CCc2ccccn2)C1)=O 22653,C1(NC(C2(OC)CCN(C(C(CC)N(C)C)=O)C2)=O)CCCOC12CCC2 22654,c1(C(=O)NCCCCN(C)C(C2CC(=O)N(O)C2)=O)coc2c(F)cccc12 22655,C1(C(=O)NCC2N(C(C=Cc3ccc(CC)o3)=O)CCC2C)CC(S(C)(=O)=O)C1 22656,CCC(CO)CCNC(=O)C(C)C(C)NC(=O)CCC1CC(C)C1 22657,C=CCC(CC)C(=O)N1C2CCC1C(CNC(=O)C=C(C)Cl)C2 22658,c1(C(=O)NCCCN(C(CCNC(N)=O)=O)C2CCCC2)nocc1Cl 22659,c1(OC)ccc(CN2CCCC(CNC(=O)C(N3CCC(OC)C3)=O)C2)cc1 22660,c1(CC)c(NC(C2CC(NCc3n[nH]c(C)c3C)C2)=O)cnn1C 22661,c1(OC)ccc(C(=O)NCC(C(C)C)NC(=O)Cc2cnn(C)c2)c(C)c1OC 22662,c1(C(N2C3C(NC(C(c4ccccc4)OC)=O)C(C3)C2)=O)ccc(=O)n(O)c1 22663,c1(C(N2C(C)CC(C(=O)OC(C)(C)C)CC2)=O)ccccc1S(C)(=O)=O 22664,C1(O)(COC)CCN(C(=O)NC2(c3cccnc3)CCCCC2)CC1 22665,c1(N2CCN(C(N3C(C)(C(=O)OC)COCC3)=O)CC2)ccnc(S(C)(=O)=O)n1 22666,CC1=C(C(=O)NC(C2CCN(C(c3ncccc3N(C)C)=O)C2)C)CCO1 22667,Cc1cccc(C(N2CC(CC(=O)N(CC(C)C(F)(F)F)C)C(C)C2)=O)c1O 22668,c1(C(=O)NC(C)(C)CCNC(c2cc(CCO)on2)=O)ccnc(F)c1O 22669,N1(C(C(C)=C2CC2)=O)CCC2(COC(CNC(C3CC3C3CC3C)=O)C2)C1 22670,C(CN=C(NCCc1nccn1C)NC1CCSC1)c1ccc(C)s1 22671,N(C(=S)NC1CCCn2c(C)nnc21)CC#C 22672,C(C)(C(C(=O)NCc1nccn1C1CC1)C(C)C)NC(C#CC(C)C)=O 22673,c1(C(N2CC(NC(c3[nH]n(C)c(=O)n3)=O)C(O)C2)=O)occ2c1CCOC2 22674,C(CNC(c1ncccn1)=O)(CC(F)(F)F)NC(=O)Cc1cscn1 22675,c1(N(CCC(=O)NC)C)nc(=NCC(CO)C2CCC2)[nH]c2cccnc12 22676,c1(NC(=O)OC)cccc(CNC(=O)NCc2nnc(-c3ccco3)s2)c1 22677,N1(C(CC(=C)Br)=O)CCC(NC(=O)COCCCC)C(F)C1 22678,c1(OC)cccc(OC)c1C(C)NC(c1cccc(F)n1)c1nnnn1C(C)C 22679,N1(C(c2cncc(C)c2)=O)CC2CC1CN2C(=O)C(C)Cc1cccc(Br)c1 22680,C1(OC)CCCC1NC(=O)CCN(C(=O)C(C)OCCOC)CCO 22681,C(=O)(C1=CCCOCC1)N1CCC(N(C(C2C3CC4C(C3)C24)=O)CC2CC2)CC1 22682,C=CCC(CC)C(=O)NC1CN(C(c2cn(C(C)C)nn2)=O)CC1(C)C 22683,C1(C2CCN(C(c3ccc(C#N)nc3O)=O)CC2)(NC(C(OC)OC)=O)CCC1 22684,c1(C(=O)NC2CC(C)(NC(CNC(CC)=O)=O)C2)cc(F)c2c(c1)CCC2 22685,C(C(=O)NCC1CC(O)CN1C(=O)C=Cc1cnccn1)(C(C)C)OC 22686,c1(CC(=O)NCCN(C(CCC(N)=O)=O)C2CCCCC2)ccc(F)c(F)c1F 22687,C(CO)(CCCNC(=O)C(c1cnn(C)c1)=O)NC(C(C)C1CCCC1)=O 22688,c1(C(=O)NC(CCNC(c2n(CC)nnc2)=O)C)cc2c(s1)CCOC2 22689,N1(C(c2ccc(C#C)cn2)=O)CCC2(CC(NC(=O)C3=NOCC3)CO2)C1 22690,c1(C(N(CCCOCCN(C(C(CC)SC)=O)C)C)=O)nc2cc(F)ccc2s1 22691,c1(C(N2CCC(C(F)(F)CO)CC2)C(=O)NC)ccc(Br)cc1OC 22692,N1(C(C(CCC)C#N)=O)CC2CCC(C(N3CCc4c[nH]nc4C3)=O)(C2)C1 22693,c1(CCCC)ccc(C(N2CC(OC)CC2C(N2C3COCC2C3)=O)=O)cc1 22694,C1(C(=O)NCCC2CCN(C(=O)CCc3ncc[nH]3)C2)CCCC(CF)C1 22695,C(CCCC(CO)NC(c1cc(C)nnc1CC)=O)NC(c1ccc(CC)[nH]1)=O 22696,C1(c2ccccc2)(SC)COCCN1Cc1cc(C)n(-c2cc(C)cc(C)c2)n1 22697,C1(C(=O)NC2CCC(CNC(c3c(C)cnnc3)=O)CC2)CCC2(C1)CC2(F)F 22698,N1(C(CCP(C)(C)=O)=O)CCOC2CN(C(=O)C=C(C3CC3)C3CC3)CC12 22699,N1(C(=O)COCCc2ccccc2)CCC2(CCCN2C(C2CCCO2)=O)C1 22700,Cc1cnsc1C(=O)NCCC1(NC(=O)C(N)=O)CCC1 22701,C1(C(=O)NCc2cc(COC)no2)CCN(C(C2(C(=O)N(C)C)CC2)=O)C1C 22702,N1(C(C(C)OCCC=C)=O)CC(O)CC1C(=O)NCCN=S(C)(C)=O 22703,c1(OC)ccc(C(C(F)(F)F)NC(c2coc(C(C)OC)n2)=O)cc1 22704,c1(C(=O)NCC2C(C)CCN(C(C)=O)C2)cc2c(c(S(N)(=O)=O)c1)CCC2 22705,C1(NC(C(C=C)(C)C)=O)CCC2(CC1)CN(C(C1(CCS(N)(=O)=O)CCC1)=O)C2 22706,c1(C(=O)OC)nc(C(=O)Nc2nc(C)c(NCCC3COCCO3)s2)oc1C 22707,N1(C(C(=O)NCC=C)c2cn[nH]c2)CC2C(OC)CS(=O)(=O)C2C1 22708,C1(CN(C(c2n(CC#C)ccc2)=O)C)CCCCN1C(c1cncnc1)=O 22709,c1(C(=O)NCCN(CCC)C(C2CCC(=O)C(C)C2)=O)cnc(C2CC2)nc1O 22710,C1(C(NCC(O)CF)=O)C(C)CCN1C(=O)C(C(C)C)SC.CC 22711,C1(N(C(CC(CC)OC)=O)C)CCN(C(=O)CCN2CCOCC2=O)CC12CC2 22712,CC(CS(=O)(=O)N=c1ccn(C2CCOC2)[nH]1)C1CC1 22713,c1(NC(c2nccs2)C(C)C)cc(-c2cccs2)n2nccc2n1 22714,C(=O)(CCC(CF)CF)NC(C(C(=O)NC(C)CC1CC1)(C)C)C 22715,Cc1cc(=NC(=O)C(C)(C2CC2)N(C)C(c2ccon2)=O)[nH]n1C 22716,c1(C(N2CC3C(NC(C(CCC)O)=O)(C3)C2)=O)cc(OC)ccc1C 22717,C12(C(N3CCC(OCCNC(C(C)n4cnnn4)=O)C3)=O)CCCCC1C2(F)F 22718,c1(C(=O)NC2CC3CN(C(CCOCC)=O)C2C3)c(F)cc(C)cc1Br 22719,Cc1nnc2cnc(C(=O)NC(C)CN(C(=O)C(C)(O)CC(C)C)C)cn12 22720,Cc1oc(C)c(C(=O)NCc2ccc(COCC(=O)NOCCCF)cc2)c1C 22721,C1(NC(CCN(C)C)=O)COCC1C(=O)NCC(F)CO 22722,c1(C(=O)NCC(C)CNC(C2CCCN2C(=O)C2CC2)=O)cncc2[nH]ccc12 22723,N1(C(Cc2cc(C)no2)=O)CCC(CNC(C2CCC(C)(C)O2)=O)C(F)(F)C1 22724,C1(CNC(CCCCNC(N)=O)=O)CCN(C(=O)CC2CCCOC2)CC1(F)F 22725,c1(OC)ccc2c(C(=O)NC3CC(C)CN(C(c4[nH]ccc4C)=O)C3)cnn2c1 22726,Cc1nc(NC(c2ccc(CCC(=O)Nc3nc(O)nc(O)n3)[nH]2)=O)cc(O)n1 22727,N1(C(CC2CC(C)C2)=O)CCC(C)(C)C(C(=O)NCC2(C)CC(C)(C)C2)C1 22728,c1(N(CCCc2cccc(C(F)(F)F)c2)C(C)C)ccc(F)cc1F 22729,N1(C2C(NC(C(CC)F)=O)CCC2)CCN(C(C2CC(O)C2)=O)CC1 22730,C(=O)(C1c2ccccc2CCN1CC(c1cc(Cl)ccc1Br)=O)OC 22731,C=C(C)CC(C(=O)NC(CCC1CCC1)C(=O)N1CC(C(C)OC)C1)OC 22732,CC1CN2CCN1C(C(N1CCCC1C1CCN(C(=O)CC3CC3(Cl)Cl)C1)=O)C2 22733,N1(C(COCCN(C)C)=O)CC(O)CCC1C(=O)NCCCc1ncn(C)n1 22734,Cc1cc(=NCc2ccsc2)[nH]c(=NCCn2cccn2)[nH]1 22735,N1(C(Cc2ccc(C)cc2Cl)=O)CCCC2CCN(C(c3oncc3C)=O)CC12 22736,c1(OCC)ccc(C)nc1C(=O)NCC1CN(C(=O)CC2COC(=O)C2)C1 22737,N1(C(CSCC#C)=O)CC2CCC1CN2C(=O)Cc1c[nH]c2ncccc12 22738,CCCC(CC)CCN1CCCC1C(N1CCCCC1)=O 22739,c1(C(=O)NC2(CC=C)CN(C(=O)C(C)CC3CCCO3)C2)cc2scc(C)c2[nH]1 22740,C=CC1(C(=O)N(CCOCC)CC)CCN(C(=O)CCCn2cccc2)C1 22741,c1(C(=O)NCC2(C)CCC(NC(c3ncn(C)c3)=O)C2)ccnc2ncccc12 22742,C12(C(N3C(CNC(c4cccc(COC)n4)=O)COCC3)=O)CC1CCC2(F)F 22743,N1(C(C2=C(C)CC2)=O)CC2COCC2(C(=O)N(C2CCCC(O)C2)C)C1 22744,O=C(CC1CCN(S(=O)(=O)c2cccc(Cl)c2)C1)N=c1cc(C2CCOC2)[nH][nH]1 22745,c1(C(=O)NCCNC(=O)C=CC(=O)N(C)C)cccc(N(CCO)CC)c1 22746,c1(CC)nc[nH]c1C(N1CCCC1CN(C(=O)C=Cc1ccsc1)C)=O 22747,c1(C(N2CC(C(=O)NCC(C)(C)C3CC3)(COC)C2)=O)ccc2cccnn12 22748,Cc1coc(C2CC2)c1C(=O)NCC1CC(NC(c2coc(CF)n2)=O)C1(C)C 22749,C#CC1CN(C(=O)CCNC(N)=O)CCN1C(C1CC1OC)=O 22750,CC1CCn2c(C(N3CC4C(NC(C56CC(CO5)C6)=O)C4C3)=O)cnc2C1 22751,Cc1ccc2occ(C(=O)NC3CCC(CNC(c4cscc4C)=O)CC3)c2c1 22752,C1(NC(C2CC=CCC2)=O)CC2(CCCN(c3c(Br)cccc3[N+](=O)[O-])C2)C1 22753,c1(C(C)C)ccccc1CC(=O)NC(C)(C)CCCNC(=O)C(C)SC(C)C 22754,C1(C(N2CC3C(C(N4CCC(C)(CO)C4)=O)(C3)C2)=O)CN2CCN1CC2 22755,c1(CC(N2CC(O)(C(C)NC(COC(C)C)=O)C2)=O)noc2cc(F)ccc12 22756,n1(CC(=O)NCCNC(C23CNC(CO2)C3)=O)cc([N+](=O)[O-])cn1 22757,N1(C(c2sc3ncn(C)c3c2)=O)CC2CCCC(C1)N(C(c1cnc[nH]1)=O)C2 22758,CCCCCC(F)C(=O)N1CC2CC1C2C(N1CCC2CC12C)=O 22759,N1(C(COc2cn(C)nc2)=O)CC(N(C)C)C(CNC(c2ncccc2N)=O)C1 22760,C1(NC(C(C)OCCOCC)=O)CCN(C(c2c[nH]cc2Br)=O)CC1F 22761,N1(C(=O)NC2CCC(N(OC)C)CC2)CCOC2(CCC(F)(F)CC2)C1 22762,N1(c2scc(CC(=O)N(C3CN(C(C4(CO)COC4)=O)C3)C)n2)CCCNC1=O 22763,c1(CCCC)ccc(C(C(=O)NCCCF)N(CCCCO)C)cc1 22764,CCCC(C(=O)NCC1(c2nn[nH]n2)CCCCC1)OCC 22765,c1(C(CNC(=O)NC(c2ccc(C)o2)CCC)COC(C)(C)C)ccccc1C 22766,CC(C)C(O)C(=O)NC1CC12CC(NC(=O)C=Cc1ccsc1Br)C2 22767,O=C(CC1=CCN(C(C2(O)CCOC2)=O)CC1)Nc1cncc(C2CC2)c1 22768,c1(C(=O)NCc2occc2C(=O)NC2CN(c3ccncc3)C2)ncc(F)cc1F 22769,c1(C(N2CCN(C(CCSC)=O)C(C)C2)=O)ccc2c(c1)nc(CO)n2C 22770,C1(C(=O)NC(CC)CNC(c2ccc(CC3CC3)cc2)=O)CC(C)(C)OC1(C)C 22771,CC1=C(C)CC(C(=O)NCCC2(CNC(C3(O)CCC(C)CC3)=O)CC2)CC1 22772,c1(OC)cc(C(=O)NCC#CCNC(=O)CCc2ccc(Cl)nc2)ncn1 22773,C1(C(N(C)Cc2ccc(Br)s2)=O)CCCN(CCC(=O)Nc2ccccc2Cl)C1 22774,CCC(CC(=O)N1CCC(CCNC(=O)C(C)(CC)OC)C1)C1CCC1 22775,CC1(C)C(NC(=O)CNC(N2CCCC2)=O)CCN1C(=O)Cc1cnccc1Cl 22776,Cc1ccn2cnc(C(=O)NCCCC3CCCN3C(C3CCCOC3)=O)c2c1 22777,C(=O)(CC(C)(C)CC(=O)N(C1CN(C(=O)C(O)c2ccco2)CC1(C)C)C)OC 22778,N1(C(C(n2ncc(C)c2)C)=O)CCC(CNC(=O)CC(C)C(F)F)C(F)(F)CC1 22779,c1(C(N(C2CCN(C(=O)C=CS(C)=O)C2)CC)=O)ccccc1Cl 22780,C1(CNC(CSCC(C)C)=O)CC2(CCC2)CN1C(=O)CC(C)n1cccn1 22781,O=C(C#CC1CC1)Nc1ncn(-c2ncccn2)n1 22782,C1(C(N2CCCC2Cn2cc(C(c3nccn3C)O)nn2)=O)(CC)CCCC1O 22783,C1(NC(Cc2nc(CC)sc2)=O)CCN(C(c2ccncc2Cl)=O)C(C)C1 22784,c1(C(=O)NC(c2ccccc2)CNC(C(C=C)O)=O)nc2ncccc2cc1C 22785,CCCC(O)CC(=O)N(C1CCCN(C(c2nccn2C(C)C)=O)C1)C 22786,C1(C(N2CC(O)(C(F)C(=O)N(C(C)C(F)F)C)C2)=O)(CC)CCOC1 22787,C1(C(=O)NCC(CN(C)C(c2ccc(CO)cc2F)=O)O)CC2(COCCO2)C1 22788,N1(C(CCCCC(=O)NC)=O)CCC2(C1)CN(C(=O)C(F)n1ccnc1)CCO2 22789,N1(CC(C)OC(=O)Nc2noc(C)c2C)CCSC(C)(C)C1 22790,S(=O)(=O)(c1ccc(=NCc2csc3cccc(F)c23)[nH]c1)N(C1CC1(C)C)C 22791,CCC(CO)(C(=O)N1CC=CC(C(=O)NOC(C)C)C1)OC 22792,Cc1cc(NC(C23CC2CCN3C(c2ccc(C)nc2O)=O)=O)c(=O)n(C)c1 22793,c1(OCC2N(C(C(=O)NC3(C)CCC3)CC3CCCO3)CCC2)ccc(F)cc1 22794,C1(CC(=O)NC(CNC(C2(COC)CCC2)=O)(C)C2CC2)C=NN(C)C1=O 22795,c1(CC=C)ccccc1C(=O)NC(C)(CSC)C(=O)NCCOC(F)F 22796,C(C(C(C)(C)C)NC(=O)Cn1c(C)csc1=O)NC(C1C(CC)C1)=O 22797,C(=O)(C(O)C(C)(C)C)N1C(C(=O)NC(COC)COC)CC2CC21 22798,C1(NC(=O)C=Cc2ccco2)CCN(C(C2(C(F)F)CCCCO2)=O)CC1CO 22799,N1(C(C2(OC)CCN(C(c3c[nH]c(C(N)=O)c3)=O)C2)=O)CC2CCC=CC12 22800,C1(CC(=O)OC)CCN(C(=O)N(C2CCN2)CCCO)CC1 22801,C1(N(c2ncncc2F)C(c2csnn2)=O)CNCC(F)(F)C1 22802,c1(CC(=O)NCC2CC(NC(c3c(=N)cc[nH]c3)=O)C2)cc(O)nc(O)n1 22803,c1(CN(C)C(c2cnn[nH]2)=O)cnn2c1CN(C(C1(CO)CC1)=O)CC2 22804,C(C)(C(=O)NC1(CN(C)C)CC1)(N(C(C(C)C1CCCC1)=O)C)C1CC1 22805,C1(NC(c2ccc([N+](=O)[O-])nc2)=O)COC2(CCN(C(C3CCC3)=O)CC2)C1 22806,C1(C(=O)NC(COC)C(C)C)CCCCCCN1C(=O)C(F)CCC(C)C 22807,c1(C(N(C2CCCC2)CC(=O)OC)=O)cc(OC)ncc1C1=CCCCC1C 22808,C1(OC)CC(NC(c2cn(C(C)(C)C)nn2)=O)CN(C(=O)CC2C=CCCC2)C1 22809,C(=O)(C(CCF)NC(=O)OC(C)(C)C)NCC(N(C(CC=C)=O)C1CC1)C1CC1 22810,C1(CNC(c2cn(CC)nc2)=O)CCC(NC(=O)CN2CCSCC2)CC1 22811,C1(NC(C2CCC(C)(C)OC2)=O)CC1C1CCN(C(c2ccoc2Cl)=O)CC1 22812,c1(NCC2(C)N(C(=O)OC(C)(C)C)CC(OC)C2)oc2ccccc2c1Cl.OCC 22813,O=C(CC(Cc1ccccc1)N1CCCC1)N1CC(CSc2ccccc2)C1 22814,c1(N2C(CN(c3snc(SC)n3)C)COCC2)ncc(C)c(C)n1 22815,c1(C(N2CCC(c3ccc(SC)s3)C2)=O)cncc(-n2cccn2)n1.C1(N)(CO)CC1 22816,CCCC(C(=O)NCC1CCC(NC(=O)C=Cc2nc(C)cs2)CC1)NC(N)=O 22817,N1(C(C(C)(C)CO)=O)CC2CC1CCC2NC(c1cn(-c2ccccc2)cn1)=O 22818,c1(OCC)ccc(-c2ccc(NC(=O)Nc3cc(C)cc(C)c3)nc2)c(C)c1 22819,N1(C(c2c(C)cccc2C)=O)CC2CCC(C1)C(NC(C1CC(F)(F)CS1)=O)C2 22820,N1(C(C2(C)CC(C)C2)=O)CCOC2(CCN(C(=O)C3=COCC3)CC2)C1 22821,C1(NC(Cn2nc(C)c(Cl)c2)=O)CCN(C(=O)CCSCC(C)C)CC1C 22822,Cc1c(C(=O)NC(CC2CC2)C(N2CC3C=CC2CC3)=O)cccc1C#N 22823,CC1CC=C(C(=O)NC(CC2CC2)C(=O)NCCn2cncn2)CC1 22824,C1(C)(C(N2CC(SCC)C2)=O)CCCN(C(=O)CC(F)(F)F)C1 22825,c1(C(=O)NCC(C2CC2)NC(C(COC)N(C)C)=O)sc(C)c(Br)c1OC 22826,C1(NC(c2c(C)nc(C(C)(C)C)s2)=O)CCCN(C(C2CCCC(C)C2)=O)C1C 22827,c1(NC(CCCCc2cccc(OC)c2)=O)cccc(SC(F)(F)F)c1F 22828,Cc1c(C(=O)NC(C)(C)C(=O)NCc2ccccc2)nc(O)c2ccccc12 22829,N1(C(CC2OCC(C)(C)C2)=O)CC2(C1)CN(C(C1(O)CCC1)=O)CCO2 22830,c1(OCC=C)ccccc1C(N1CCCC1(C)C(=O)NCc1ccccn1)=O 22831,C1(CNC(C=CC(C)=O)=O)CC2CCC(C1)N2C(=O)CCCc1cccnc1 22832,Cc1ccc(C(F)C(N2CCCCC2CCNC(=O)CSCCC#N)=O)cc1 22833,C1(CNC(=O)C(O)Cc2cnc[nH]2)C2CN(C(C3CC(F)(CF)C3)=O)CC12 22834,C1(C(=O)NC)CCN(C(C2(CSC)CN(C(c3ccn(C4CCC4)n3)=O)C2)=O)C1 22835,N#Cc1c(Cl)ccc(NC(C2CN(Cc3ccnc(O)c3)CC(F)(F)C2)=O)c1Cl 22836,C1(NC(c2cnn(CC(F)F)c2)=O)CCC(O)CN(C(=O)CC2CCNC2=O)C1 22837,c1(C(=O)NCC(CNC(Cc2c(C)n(C)cn2)=O)C)ccc(S(N)(=O)=O)nc1 22838,CC(CC(C)(C)C)C(=O)NCc1ncc(C(=O)NCC2(O)CCN(C)C2)cn1 22839,C(CNC(=O)NCc1cc(C)c(F)c(C)c1)(CCS(C)(=O)=O)OC 22840,N1(C(C2CN(S(CC)(=O)=O)C2)=O)CCCC(CO)(NC(C2COC(=O)N2C)=O)C1 22841,C1(CC)CN(C(c2c(C)nnn2C)=O)CCC1NC(=O)C(C)(C)CN(C)C 22842,c1(C(N(CC(CC)NC(C=CC)=O)CC)=O)cnn2cccc(Br)c12 22843,N1(CC(=O)NC2C(NCC(=O)NC3CC(C(F)F)C3)CCC2)CCOCC1 22844,C1(CN(C(=O)CCCNC(C)=O)CC)CCN(C(c2cc(C)cs2)=O)CC1 22845,CC1CCc2sc(C(=O)NCC3CCCN(c4nc5ccccc5o4)C3)cc2C1 22846,c1(NC(C(c2cc(C(=O)OC)ccn2)N(CC=C)CC#N)=O)ccc(F)cc1C 22847,C(=O)(CC(O)C(C)C)NCC1(C(=O)N(CCCF)C)CC(=C)C1 22848,C1(CN(C)Cc2cnn(C)c2)CCN(C(=O)C(C2CCOCC2)=O)CC1 22849,C(=O)(C1=CNC2=NCCCN12)N1CCCCC(NC(C2CC(C)N(C)C2)=O)C1 22850,C1(CNC(C(C)C2CC2)=O)CN(C(=O)Cn2ncc3ncccc23)CCC1(C)C 22851,c1(C(N2CCC(C3N(CC#C)CCC3)CC2)=O)cc(C#N)[nH]c1C 22852,C1(C(N(C)CC2(CC(C)C)CC2)=O)CC2(CCN(C(C3CCCCS3)=O)C2)C1 22853,C(=O)(C(C)CC(=O)NCCCc1cncc(C(=O)OC)c1)OC 22854,c1(NC(C(=O)N(C)Cc2c(OC(F)F)cccc2Cl)=O)cccc2c1CCC2 22855,c1(C(C)(C)C)nc(=NCC2CCCCN2C(=O)Cn2cncn2)s[nH]1 22856,C1(NC(c2cc(C)ncc2)=O)CCN(C(C2OCCCO2)=O)CC1F 22857,c1(C(N2CCC(N(C(C)=O)C3CC3)C2)=O)c(Cl)cc(Sc2nnc(C)o2)cc1Cl 22858,CCC(C)C(C)C(=O)N(C)CC1CCCCN1C(=O)C(C)CC1CCCC1 22859,CC(C)(C(=O)NCC1CN(C(C2CCS2(=O)=O)=O)C1)c1ccccc1 22860,Cc1cc(CC(N2CCC(O)(c3cc[nH]n3)C2)=O)ccn1 22861,n1(CC(N2CCCC(N(C(C3CC3CF)=O)CC)C2)=O)cc([N+](=O)[O-])cn1 22862,Cc1cc(Cl)c(C(=O)NC2CC3CC(NC(C4C5(CC5)C45CC5)=O)C3C2)cc1C 22863,Cc1ccc(C(N2CCCC(C)C2CNC(=O)C(F)F)=O)cc1[N+](=O)[O-] 22864,c1(C(N(CC(C)(C)NC(CC(=C)Br)=O)C)=O)ccc(C(F)(F)F)nc1C 22865,Cc1nc2nccc(C(=O)NC3CCCC(CNC(C4CN(C)C4)=O)C3)n2n1 22866,N1(C(=O)C2=C(Cl)CCC2)CCC2(CCCN2C(C2CC3(C2)CC3F)=O)C1 22867,c1(C(N2CCOC(C)(C)CC2)C(=O)NCC=C)cccc2ccsc12 22868,Cc1ccncc1C=CC(=O)NC1CC(NC(=O)C(=C2CCCCC2)F)CC1O 22869,CC(CCCCNC(C1CCOC1C1CC1)=O)NC(c1ccc(F)nc1)=O 22870,C(=O)(C1=C(C)C(C)(C)OC1=O)N1C(COC)CN(C(=O)Cc2ccc(C)s2)CC1 22871,C1(C)(CNC(c2c(C)cc(Cl)cc2)=O)CN(C(=O)C(=O)N(C)C)C(C)(C)C1 22872,C1(C(N(CCN(C(=O)CC2CCC(=O)N2)C(C)C)C)=O)CCNC(=O)C1 22873,N1(C(CCC(C)C)=O)CCC2(CCCCN(C(C3(C(F)F)CC4(CC4)C3)=O)C2)C1 22874,C1(C(=O)NCC(C)(C)NC(C(C)NC(c2ccco2)=O)=O)C(C)(C)OC1(C)C 22875,CCCC(CC(C)C)C(=O)N1CC=CC1C(=O)NCC(=O)OC 22876,c1(NC(CCC(=C)C)C)ccc(S(=O)(=O)NCc2csc(C)n2)cn1 22877,C1(C(=O)NCCC2COCCN2C(c2cnc(SC)n2C)=O)(CC)CC(C)(C)C1 22878,Cc1nc2cncc(C(=O)NCC3CN(C(C4C(Cl)(Cl)C45CC5)=O)CCO3)c2[nH]1 22879,C(=O)(C1=NOC(C)(C)C1)NCC1(NC(C2C(c3c(C)cccc3)C2)=O)CC1 22880,C(=O)(CCCc1ccncc1)N(CC(CC)NC(=O)C(C)(C)C1CC1)C 22881,N1(C(C(C)(C)CF)=O)CCC2(CCCC2CNC(c2ccnc(O)c2)=O)CC1 22882,S(=O)(=O)(c1c[nH]c(C(=O)NCC2CC(C)N(C(C3C4(CC4)C34CC4)=O)C2)c1)NC 22883,CC1CCN(C(c2cccn3ccnc23)=O)C(C)C1NC(c1nn(C)cc1Cl)=O 22884,N1(C(C2(C=C)CCC2)=O)CCCC(CC(=O)NCCC2CCCN2C)C1 22885,c1(C(=O)NCC23N(C(COCCOC)=O)CCC2CC3)nccn2nccc12 22886,C(=O)(C1=Cc2ccccc2OC1)N(CC(C)NC(=O)C(N1CCCCC1=O)C)C 22887,c1(OCCCC)ccc(C(=O)NCCCc2cn(CCC(F)(F)Cl)nn2)cc1 22888,c1(C(=O)NC2C(C(N)=O)CN(C(C3CC3(F)F)=O)CC2)ccc2c(c1)OCO2 22889,c1(C(C)=O)cc(O)cc(O)c1C(=O)NCC12CC1CN(C(c1cc[nH]n1)=O)C2 22890,c1(OC)cc(CN2CCC(C(=O)Nc3ncn(C)n3)C(O)C2)c(Br)cn1 22891,c1(C(=O)NC2C(NC(C3(CCCC)CCCC3)=O)CC2)cnc2[nH]cnc2c1 22892,C(CNC(C1(C(F)F)CC1)=O)(C(C)C(C)C)NC(c1cc(C)c(C)[nH]1)=O 22893,N1(C(C2CCC(C)O2)=O)CC=C(CCNC(c2cc(Br)n[nH]2)=O)CC1 22894,C1(CC(=O)OCC)CC(F)CN1C(=O)CCCCc1cn(-c2ccncc2)nn1 22895,N1(C(c2cn(CC)nc2)=O)CCC(C)(C)C1CC(N1CC(C)(C#N)C1)=O 22896,S(=O)(=O)(c1cccc(-c2nnc(CN(C)C)o2)c1)N(C)C1CC1 22897,C1(NC(c2c(C)cco2)=O)CN(c2nnc(CC(C)C)s2)CC2(CC2)C1 22898,C(C1C(C(=O)N(C)CCOCCNC(c2sc(CO)nc2C)=O)C1(C)C)=C(C)C 22899,O=S(c1ccc(NC2CCc3c(O)cccc32)cc1)C(F)(F)F 22900,c1(C(=O)NC2CC3(CN(C(C4(SC)CC4)=O)C3)C2)cc2nc[nH]c2cn1 22901,CCC(CC)C(F)C(=O)NCc1nnn(C)c1C(=O)N(C1CC2CC2C1)C 22902,C1(C(=O)NC(C)C(=O)N(C)CCN(C)C(C2CC(O)C2)=O)CCCCC1 22903,Cc1ccc([N+](=O)[O-])c(C(=O)NC2CCCN(C(c3c(C)nsc3C)=O)C2)c1C 22904,CCC(CC)CCCC(=O)NCC1(O)CCN(C(c2noc(C(C)C)c2C)=O)C1 22905,C1(NC(c2csc(Cl)n2)=O)CC(O)CN(C(c2ccc(OCC3CC3)nc2)=O)C1 22906,C12(CNC(C(CC=CC)C)=O)CCCC(CN1C(=O)Cc1cnccc1Cl)C2 22907,N1(C(C(CCC)(C)O)=O)CC(=O)NC2(CCOCC2)C1 22908,C1(NC(C2(N=[N+]=[N-])CC2)=O)CCCN(C(c2cc(C(F)(F)F)cs2)=O)C1 22909,C=CCC(C)(C)CC(=O)NC1CCC(N(C)C(c2cc3ncccc3s2)=O)CC1 22910,C1(NC(c2nc(C)sc2)=O)CN(C(C2C=CCC2)=O)CC12CCS(=O)(=O)CC2 22911,C(=O)(C(O)C1=CCCCC1)N1CC(C)(OCC(N2CC3CCCC2C3)=O)C1 22912,C1(C(=O)NC2CC(CN=c3nc(C)[nH]s3)C2)CCc2ccccc2O1 22913,C1(C(=O)NC(c2cn[nH]c2)C)CCN(C(c2cnnn2C)=O)CC1 22914,N1(C(C(CO)OC)=O)CCC2(CC1)CC(NC(=O)CCCn1ccnc1)CO2 22915,c1(OC)c(CC(=O)NC(C2CCCC2)CNC(=O)C=CCF)cccc1Br 22916,C(CC(=O)NCC1CCN(C(C)=O)C1)(C(C)C)NC(c1ccn(CC)c1C)=O 22917,c1(C(=O)NCC2CN(C(C3C(CCOC)C3)=O)C2)ccc(O)c(CC(C)C)c1 22918,C(C)(N=c1cc(C)nc(N2CCC(CC(C)C)C2)[nH]1)c1[nH]nc(C(=O)OCC)n1 22919,N1(C(c2ccc(CN(C)C)o2)=O)CCC(CO)(CNC(C2CCS(=O)(=O)C2)=O)C1 22920,c1(CC)cc(CNC(=O)C(C)=CCNC(c2cc(OC)n[nH]2)=O)on1 22921,CCC(C)(C)C(C)NC(C1CCN1C(=O)C(C)NC=O)=O 22922,C=CC1OCCC1C(=O)NCCC1CC(NC(=O)CCC2CC2C)C1 22923,c1(OCC)cc(Cl)ccc1C(N1CCN(C(=O)CCC=CBr)CC1CF)=O 22924,Cc1cn(C)nc1C(=O)NC(CC1CCCC1)C(=O)NC1CCOCC1F 22925,C(=O)(C1COc2ccccc21)N1C(CNC(c2n[nH]c(C)c2O)=O)CC(F)(F)C1 22926,CC(C)C(O)C(C)C(=O)NCC1CCOC1C(N1CC2CC(O)CC1C2)=O 22927,N1(C(=O)OC(C)(C)C)CCC2CN(C(=O)Cc3ncc(Cl)s3)C2C1 22928,C(=O)(CC(O)CC(C)C)N1CCN(C(C(CCCOC)C)=O)CC1c1ccco1 22929,c1(NC)c(C(=O)NC2CN(C(=O)CCSc3nccn3C)CC2O)cccc1F 22930,c1(C(=O)NC2C(NC(=O)CC3CC4(CC4)CO3)CCC2)ccc2c(c1)CNC2=O 22931,C#CCCC(O)C(=O)N1CC(F)CC1CNC(C1(S(N)(=O)=O)CC1)=O 22932,c1(C(=O)NC2C(F)CCN(C(C3CC(=C)C3)=O)C2)ccc2nc(C(F)F)[nH]c2c1 22933,C1(C(=O)NC(CC#C)CC#C)CCCCCN1C(C1CC(C)=NO1)=O 22934,c1(C(=O)NCC(C(C)(C)C)NC(C(C)OCC#C)=O)ccc(C#N)c(O)c1 22935,N1(C(c2nn(CC)c(O)c2)=O)CCCC(C)(C)C1CNC(=O)C(C)(C)OC 22936,c1(C(=O)NCC2(F)CN(C(C3C4CCOCC34)=O)C2)ccc2ncnc(O)c2c1 22937,CCCCCCCCCCCCCCCOC(C1CC(=O)NC2(CCC2)C1)=O 22938,c1(CNC(C2CCC(F)C2)=O)ncc(Cl)cc1Cl 22939,c1(-n2cnc(C(N3CCC(NC(CCC=C)=O)C3)=O)n2)ncccc1F 22940,N1(C(CSC(C)=O)=O)CCc2[nH]nc(C(=O)Nc3cc(Cl)c(O)c(Cl)c3)c2C1 22941,c1(C(=O)NCC(=O)NC2CC(C(=O)NCC3CCCC3)C2)cc(C(F)(F)F)on1 22942,Cc1oc(CNC(C2CN(C)C2)=O)nc1C(=O)N(C)CCC1CCC1 22943,c1(C(=O)NCC2(CN(C)C)CCC2)ccccc1-n1cc(CCS(N)(=O)=O)nn1 22944,C12(C(N(CC(CCC)C)C)=O)C(NC(c3cocn3)=O)C3CC1C2C3 22945,N1(C(CO[Si](C)(C)C)=O)CC(O)CC1CNC(C1(C(F)(F)F)CC=CC1)=O 22946,C12(COC)CC(C(=O)NCC(C3CCCN3C(=O)C(C)CN(C)C)(C)C)(CO1)C2 22947,C1(CC(=O)NCC(O)C2(Cl)CC2)CCCN1C(c1cnsn1)=O 22948,c1(OCC)cc(CNCCc2noc(C3CCOCC3)n2)cc(F)c1 22949,Cc1nnn(CC(=O)NC(C)C(=O)NCc2ccn(C3CC3)n2)n1 22950,N1(C(C(C)(C)NC)=O)CCC2(CC1)CC2NC(c1cnn(CCCOC)c1)=O 22951,c1(CC)nc[nH]c1C(=O)NCC1(Cn2cc(C(C)OC)nn2)CC1 22952,Cc1csc(Cl)c1C(=O)NCC1CN(C(=O)CC(c2cccc(F)c2)O)CC1C 22953,c1(C(=O)NC2CCC(CC(=O)NC3(CC)CC=CC3)CC2)cc2ccccn2n1 22954,Cc1nnc2n1CC(NC(=O)C(F)C1CCOC1)C2 22955,c1(C(=O)Nc2c(CC(=O)OCC)nccc2)nn(C)c2ccc(Br)cc12 22956,CC(C)CC(C(=O)N1CCCC(CNc2ncccc2C#N)C1)C(N)=O 22957,N1(C(c2occ(C)c2)=O)CC2OCCN(C(C3CCCCS3(=O)=O)=O)C2C1 22958,N1(CCOCC)CCc2c(NC(c3cc(CC(F)(F)F)ccc3F)=O)cccc2C1 22959,N1(C(CCCCC)=O)CC2(C1)CN(C(=O)CCC1CCCC(O)C1)CC2CO 22960,C(=O)(C(CCCC)C(C)C)N1CCC(C(=O)NCCOCC=C)C1CC 22961,C1(C2(NC(c3c(CCCC)ocn3)=O)CC2)CCCCN1C(=O)C=CC(F)(F)F 22962,Cc1cn2c(n1)CC(C(=O)NCC1CC3(CC3)CN1C(c1cnsc1)=O)C2 22963,CC1(C)C(NC(=O)CCSc2ccc(Cl)cc2)CCN1C(=O)C(O)CC1CC1 22964,N1(C(CCC(C)C)=O)CC(C)CN(C(c2cccc(C(C)(C)C)c2)=O)C(C)C1 22965,c1(C(=O)NC2C(NC(C3=CCCC3C)=O)C2)cc2c(s1)CCCCCC2 22966,N#Cc1ccc(NC(C2CN(C(c3cccc(Cl)c3)=O)CC(F)(F)C2)=O)cc1Cl 22967,N1(C(CC=C)=O)CCC(N(C)C(C2CCN(c3cnn(C)c3)C2=O)=O)C2(CC2)C1 22968,C(=O)(C(CCC(C)C)NC(C1CN2CCN1CC2)=O)N(CC(=O)OC)CC 22969,CC(O)CCC(=O)NC1CCC(N(C(=O)CCc2ccccc2C(N)=O)C)CC1 22970,C1(CC#C)(C(=O)NC2CCC2NC(C2CN(c3nncs3)C2)=O)CCCCO1 22971,C1(C)(COC)CC(NC(c2cc(N)ccc2Cl)=O)CN1C(=O)CCCC1CC1 22972,c1(C(C(=O)NC2C(NC(c3occ(C(=O)OC)c3)=O)CC2)O)ccc(F)cc1C 22973,CC(C)CC(C(=O)NCC1CC(C)N(C(=O)COC(C)C)C1)C(N)=O 22974,C(=O)(CC(C)c1ccncc1)N(CC(C)O)CCNC(=O)CCSC(F)(F)F 22975,Cc1ccc(C(=O)NC2CN(C(C3CC(n4cnnc4)C3)=O)C2)cc1Cl 22976,c1(C(=O)NC(CNC(C(CCC)C)=O)C(C)C)c(NC(=O)C2CC2)sc(C)c1C 22977,c1(C(=O)NCCN(C(C23COCC2C3)=O)CC2CC2)sc2sccc2c1Cl 22978,CCCCC(CNC(c1cc(C#N)c[nH]1)=O)NC(=O)COCC1CCOC1 22979,c1(C(N2C(C(C)C(=O)O)CCC2)=O)cc(C(F)F)ccc1Br 22980,CC1=C(C(=O)NC2CC2CNC(C2(C)CCC2)=O)CCCC1 22981,N1(C(C(COCC)C)=O)CC(N(C)C(c2cnc(SC)nc2O)=O)C2(CC2)C1 22982,c1(OC)cc(NC(c2cnc(F)c(C)c2)=O)c(OC)cc1Br 22983,c1(C(c2n(CCOC)nnn2)NCC(c2cccs2)C2CC2)nc(C)c(C)[nH]1 22984,CC1CCN(C(=O)CN(C)C(=O)C2CC2)CCN1C(C1C2CCN1CC2)=O 22985,c1(CNc2c(C(=O)NCC)nccc2)oc2ccccc2c1C 22986,C(c1ccc2c(c1)COCC2)=CC(N1CC2CCN(C(CC(C)C)=O)CC2C1)=O 22987,N1(CC(N2CCCCCC2)=O)CCC2CC(NC(c3ccc(C)s3)=O)C2C1 22988,C1(C2CCC2)(C(=O)NCC2(C(C)(C)C)CCN(C(c3cnns3)=O)C2)CC1 22989,N1(C(c2c(C(C)C)nn(C)c2)=O)C(CNC(=O)COCC2CC2)CC2COCC12 22990,c1(C(N(C(C)CNC(=O)CC2CCC2)C)=O)ccc2c(c1)CCN2C(C)(C)C 22991,CC12CC(C(N3CCC(F)(CNC(=O)C4=CCCOC4)C3)=O)(CCO1)C2 22992,C1(C(N(C(C(C)C)C)C)=O)CCN(C(=O)CCCc2cnn[nH]2)CC1O 22993,N#CC1(C(=O)NCC2(CNC(=O)CN3CCCC3CO)CC2)CC2(CCC2)C1 22994,C(C)(C)(CCC(=O)N1CCCC(COC)(NC(=O)Cc2ccco2)C1)OC 22995,C12(C(=O)NCC3CN(C(C4CCCC45CCC5)=O)CCO3)C3CC(CC13)C2(F)F 22996,c1(C(=O)NCCOC2CN(C(C3C(C)C3C)=O)C2)csc(Cl)c1 22997,N1(C(C2(C)CCCN2)=O)CCCC2CN(Cc3noc4c3COCC4)CCC12 22998,C=CC(C(=O)NCCC1(O)CN(C(=O)C(C)SC)C1)OC 22999,CC(C(=O)N1CCC(C(C)C(=O)NCCc2nncs2)C1)C(F)F 23000,C(C1c2ccccc2CCN1C(=O)COC1CC1)NC(C1CCCS(=O)(=O)C1)=O 23001,Cc1ccc(F)cc1CC(=O)NCCCC1CCCN1C(C1C2CCC1CC2)=O 23002,C(=O)(C(C)(O)CCN(C)C)N1C2C(CNC(CSc3n(C)cnn3)=O)C(C2)C1 23003,C1(C(N2C(CN(C(c3c(CC)non3)=O)C)CCCC2)=O)Cc2ccncc2C1 23004,c1(OC)cc(C(N2CCC(OC)C2)=O)ncc1Cc1ccccc1 23005,S(=O)(=O)(c1ccc(F)c(F)c1)N1CCC(NC(c2ccc(C(N)=O)nc2)=O)C1 23006,Cc1cc(O)ncc1C(c1nnnn1C)NCCCSCCC(F)(F)F 23007,CC1(C#N)CCN(C(=NC2CCC2)NC2CC(OC(F)F)C2(C)C)CC1 23008,CCC(C)C(O)C(C)C(=O)NC(Cc1ccco1)C(N1CCC(O)(CO)C1)=O 23009,c1(C(N2CCC(C3(NC(C4CC4(F)F)=O)CC3)C2)=O)ccc2ncccc2n1 23010,N1(C(c2n[nH]c(CC)c2Cl)=O)CCCC(O)(CNC(C2CC23CC3)=O)CC1 23011,N1(C(c2c(CC)cno2)=O)CC(N(C(=O)C(C)NC(C)=O)C)C2(CC2)C1 23012,N1(C(C=CC(=O)OCC)=O)CCN(C(c2coc(Br)c2)=O)C(CF)C1 23013,c1(CC(N2CC(CNC(C(C)C)=O)OCC2)=O)ccc2ccncc2c1 23014,CCCC(C)(O)CNC(C1(CNC(=O)Cn2ccc(C)n2)CC2(CC2)C1)=O 23015,C1(NC(CP(C)(C)=O)=O)CC2CCC1(CNC(=O)CN(C1CCC1)C)C2 23016,C1(NC(c2ccc(OC(F)F)cc2)=O)CCN(Cc2nccc(C(F)F)n2)CC1 23017,c1(SC)ccc(CN(C(c2cc(C)ns2)C(=O)NCC2CCCO2)C)cc1 23018,C=C(CNC(=O)C(C)(C)C1CCCC1)CCNC(=O)CSCCOC 23019,C(C(=O)N(C1CCN(C(C2(OC)CCCC2)=O)C1)CC)(C(C)C)SCC 23020,C1(CNC(C(CC=CCC)C)=O)CN(C(c2cc(Cl)nn2C)=O)CC1(F)F 23021,c1(C(=O)NCCC2CN(C(C3CCCS3)=O)CCO2)coc2c1COC2 23022,N1(C(c2cn(CC=C)nc2)=O)CC(O)CC1CNC(=O)C(C)OCCOC 23023,Cc1nc2[nH]c(C(N3CC4CCC(NC(=O)CCNC(N)=O)(C4)C3)=O)cc2s1 23024,N1(C(C(C)N(CC(F)(F)F)C)=O)CCC2(CC1)CC2CNC(=O)CN1CC(C)(C)C1 23025,Cc1cc(NCCc2ncc(Br)cn2)ncc1S(=O)(=O)NC(C)(C)C1CC1 23026,C1(NC(C2C(NC(Cc3n(C)ccn3)=O)COC2)=O)CCCCC12CC2 23027,N1(C(c2cc(OC)nc(F)c2)=O)CCN(C(c2c[nH]nc2C(C)C)=O)CC(O)C1 23028,c1(SCCC(CNC(=O)NCC2C(COC)C2)C(=O)O)ccc(F)cc1 23029,C1(CNC(=O)CC2=CCCC2)CC2CCC1N(C(=O)CC1CCC3CC13)C2 23030,N1(C(c2c(-c3cn(C)nc3)onc2)=O)CC=C(CCNC(c2ccsc2)=O)CC1 23031,C1(O)(C(C)NC(C(C)OCC=C)=O)CN(C(=O)C=Cc2ccc[nH]2)C1 23032,c1(C(=O)NCCCC(=O)OC)ccccc1NC(=O)Cc1ccccc1 23033,c1(C(N2CCCC(CCNC(C(CN(CC)CC)F)=O)C2)=O)cnc(O)cc1O 23034,c1(C(N2C(CN(C(C(CSC)(C)C)=O)C)COCC2)=O)nsc2ccc(C)cc12 23035,c1(NC(C2CC2C(=O)Nc2ccc(C3CC3)cc2)=O)cncc(C2CC2)c1 23036,c1(SCCCNC(=O)Nc2nnc(-c3c(F)cccc3F)s2)cc2c(s1)CCC2 23037,CC1CCC(C)N1CC(=O)NCCc1ccc(C(=O)N(C)C)cc1 23038,c1(C(N(C)CCN(C)C(C2(C#N)CC2C(F)(F)F)=O)=O)cccc(F)c1F 23039,N1(CCC(=O)NC2CC(C)(NC(C3C=CCCC3)=O)C2)CCCS1(=O)=O 23040,c1(C(=O)NC2CC3CC(NC(C(CN(C)C)O)=O)C2C3)cc2ccccc2o1 23041,Cc1cccc(-c2cc(C(=O)NCC(C(C)C)NC(=O)C(C)(C)C3CC3)on2)c1 23042,c1(C(=O)NC2(C)CC(NC(C(C)(C)NC(=O)OC)=O)C2)cc(OC)cc(Cl)c1F 23043,C1(C(N(CC(CN(C(=O)CC2CC(F)(F)C2)C)O)C)=O)CCC(F)(F)CC1 23044,CC(C)CC(F)C(=O)NCC1C2CCC(C2)N1C(C1CCN(C(=O)N(C)C)CC1)=O 23045,c1(OC)cc(F)cc(C=CC(=O)NC2CCC2NC(=O)C2=CCCCCC2)c1 23046,CCC(C)(CCNC(c1nocc1C)=O)NC(=O)COC1(C)CCCC1 23047,N1(C(c2cc(SC)ncc2)=O)CCCC(C2CC2NC(C2CC=CCO2)=O)C1 23048,c1(CN(C(=O)C(C2CCC2)NC(C2C=CCS2)=O)C)ncc[nH]1 23049,C(=O)(CC(C)(C)O)NC.C(=O)(C(C)OCCC(C)C)NC1(CC(=O)OC)CC1 23050,N1(C(CC(C(C)(C)NC(C2C(C)CC2)=O)C)=O)CCc2ncccc2C1 23051,N1(C(CC2CCC(=O)NC2)=O)CC2CC3CC2C1C3NC(C1CCC2(CC2)C1)=O 23052,CC(C)(O)C(C(=O)NOC1CC1)NC(c1ccc(=O)n(C)c1)=O 23053,C(=O)(C(O)CCCC)NCCC1OCCN(C(C2(C=C)CC2)=O)C1 23054,N1(C(C(F)=CC)=O)CCC2CN(C(C3CCN(c4ccccc4)C3)=O)C2C1 23055,C1(C(N(C(C)CNC(C2(CCF)CC2)=O)C)=O)CCC(NS(C)(=O)=O)C1 23056,c1(NCc2cc(C)cc(N)c2)cc(Br)ccc1S(=O)(=O)N1CCCNC(=O)CC1 23057,N1(C(c2n[nH]cc2Br)C(=O)NCc2cccc(OC)c2)CCNC(=O)C1CCO 23058,C12(C(C)NC(C3(C)CC3)=O)CC(NC(C3CN(CC(F)F)C3)=O)(C1)C(C)O2 23059,c1(C(CC(=O)NCc2ccc(COC(C)C)cc2)C)ccc2c(c1)OCO2 23060,C1(OC)CN2CCCC2(C(=O)NCC2CC(NC(c3c(Cl)cccc3Cl)=O)C2)C1 23061,N1(C(C(C)=CC)=O)CC2CN(C(c3cccc(NC(=O)OC)c3)=O)CC2C1 23062,N1(C(C=C(CC)CC)=O)CC(CNC(C2(CO)CCOCC2)=O)C2(CCC2)C1 23063,N1(C(C2C(CNC(C3CCCS3)=O)CC2)=O)CC(F)(F)C(F)(F)C1 23064,C#Cc1ccc(C(=O)NC2CN(C(=O)Cc3sc(O)nc3O)CC23CC3)cc1F 23065,CC1CCC=C1C(=O)NC1CCCC(C(=O)Nc2cnn(C)c2Cl)CC1 23066,Cc1ncnc(C(N2CCC(NC(=O)CC3C=CCCC3)C2C)=O)c1C 23067,C1(NC(CC)=O)(CNC(C2CCN2S(C)(=O)=O)=O)CCC(C)(C)CC1 23068,C1(O)(CC(N)=O)CCN(C(c2ccc(O)nc2)C(=O)Nc2ccccc2Cl)CC1 23069,c1(C(N2C(CNC(C3N(C)CCCC3)=O)CC(O)C2)=O)ccc(N)c(Cl)n1 23070,C1(CN(C(CC(=O)OCC)=O)C)CN(C(C2(C)CCN(C)C2)=O)CCO1 23071,c1(C(=O)NCc2cn(C3CCN(C(C=C(CC)C)=O)C3)nn2)ccccc1C 23072,Cc1cc(N2CC(F)(F)CC2CNC(=O)C(c2cccnc2)O)n2ncnc2n1 23073,S(=O)(=O)(c1ccccc1Cl)NCCC(=O)N(C)CCNC(c1ccns1)=O 23074,c1(CC(N2CCN(CC3CCCN(C(COC)=O)C3)CC2)=O)csc2nccn12 23075,S(=O)(=O)(c1cccc(=NCC(C)c2cccs2)[nH]1)NCCCCCC(=O)NC 23076,N1(S(CCOC)(=O)=O)CCC(N=c2nc[nH]n3cc(Br)cc23)C1 23077,C1(NC(c2ccn(C(C)C)n2)=O)CC(CNC(c2cc(C(N)=O)cs2)=O)C1(C)C 23078,C1(CNC(c2cccc(C)n2)=O)CN(C(=O)C(C)(C)C2CCCO2)CCN1C 23079,C1(C(C)C)CCC(NC(c2nc(NS(=O)(=O)CCBr)cn2C)=O)CC1 23080,C1(NC(CCCCCC)=O)CC2CN(C(c3cc(C)n(C(C)(C)C)n3)=O)CC2C1 23081,c1(C(=O)NCC2OCCCN(C(C(C(C)C)F)=O)C2)ccc2c(c1)C(C)(C)CO2 23082,C1(S(N)(=O)=O)(C(=O)NCCCNC(C2(C(=O)OCC)CC2)=O)CC1 23083,C(=O)(CC(C)CNC(C1CCC(=O)N1)=O)NCc1nnc(CC)s1 23084,C(CO)(C(F)(F)F)NC(C(Cc1cc[nH]n1)NC(=O)CCn1cncn1)=O 23085,N1(C(C=C(C)c2cccs2)=O)CCN(C(c2ccc3cc[nH]c3n2)=O)CCC1C 23086,C1(C(N2C(CNC(c3ncoc3C(F)(F)F)=O)CCC2)=O)CCC2(CCC2)C1 23087,c1(OC)cccc(C(N2CCC(CF)(NC(=O)Cn3cccn3)C2)=O)c1 23088,c1(NC(C2(C)CCN2C(c2cnc(C3CC3)nc2)=O)=O)nc(Br)ccc1Cl 23089,N1(C(CC(C(C)C)O)=O)CC(C)(CNC(=O)COCCCN(C)C)CC1(C)C 23090,C#CCCCCC(=O)NCC(CC(=O)NCC(=O)OC(C)C)C1CCC1 23091,N1(C(CCC)=O)CCN(C(c2[nH]ccc2C2CC2)=O)CC1CC1CC1 23092,Nc1ccc(NC(N2CC(CC(=O)C(=O)O)C2)=O)cc1Cl 23093,CN1CC=C(C(=O)NC(CC2CCCC2)C(=O)NC2CCCN(C)C2)C1 23094,C1(C(=O)NCCC2CCN(C(=O)C(C3CCC3)C3CCC3)C2)CC(F)C(=O)N1 23095,c1(CNC(c2cc(CC)on2)=O)ccc(CNC(C2(C)COC2)=O)cc1F 23096,C1(CC(=O)NCC(C)NC(c2nnc(C(C)(C)C)o2)=O)CCOCC1 23097,c1(SC)cc(F)ccc1C(=O)NCCOCCNC(=O)COCC(F)F 23098,C1(N(C(CSC)=O)CCO)CCN(C(c2cc(CSC3CCC3)c[nH]2)=O)C1 23099,N1(C(C(CC)O)=O)CCN(C)CC1C(=O)NOCC(F)F 23100,CN1CC(NCCc2c[nH]c3cc(F)ccc23)CCc2ccccc21 23101,c1(OC(C)C(=O)NCC2(O)CN(C(=O)Cn3cnnn3)C2)cccc(Br)c1 23102,c1(C(N2CCC(N(C(c3coc(O)n3)=O)CC)C2)=O)cc(F)c2ncccc2c1 23103,c1(C(=O)NC(C)C(C)(C)NC(=O)CCNC(c2ccsc2Cl)=O)ncc(F)cn1 23104,Cc1ccc(C2CC2NC(C2CC(C)CCN2C(=O)C(O)C(F)(F)F)=O)c(Cl)n1 23105,c1(C(N2CC(NC(C3C(C(C)C)C3)=O)C3(C2)CC3)=O)cc(Cl)cc2ccncc12 23106,N1(C(CCCOC(C)C)=O)CC2(CC(NC(c3csc4cncn34)=O)C2)C1 23107,C1(N(C(C2C(OCC)C2)=O)CC)CCN(C(=O)Cc2cccc(F)c2)CC1 23108,N1(C(c2cc(C)on2)=O)CCC2(CCC(NC(=O)CCP(C)(C)=O)C2)C1 23109,CN1CC2C3CCN2C2C=CC(=CC=C1N1C(=O)N=C3C1=O)CC(CC)CC2 23110,C(CN=c1nc2scnc2c(NCC2CC2C2CCCC2)[nH]1)N(C(=O)OC)C 23111,Cc1ccc(C(O)C(=O)N(c2cnncc2C)C2CC3(CNC3)C2)nc1 23112,c1(C(=O)NCC2C(C)CCN(C(C34CC(C)(C3)C4)=O)C2)ccc2nn[nH]c2n1 23113,c1(C(N2CCCN(C(C3CC4CCC3O4)=O)CC2)=O)ncc(F)cc1F 23114,n1(C(C)C)cc(C(=O)NCCCN(C)C(C2CC2c2ccsc2)=O)nn1 23115,N1(C(c2c(OC)cc(F)cc2)=O)CCCN(C(=O)CC(C)C)C(C)C1 23116,C1(NC(=O)Cc2cnc[nH]2)CC2CCC1CN(C(C1CCOC1C(F)(F)F)=O)C2 23117,c1(N2CCCC(SCC(=O)Nc3ccc(C)cc3)C2)cc(C(=O)O)c(Br)cn1 23118,C1(C(=O)NCC2C(CNC(Cn3ccc(C)c3)=O)C2)CCC2(CC2)C1 23119,C1(OCC)CC2(C1)CC2NC(C1C=CCN1C(C1CCC1COC)=O)=O 23120,N1(C(C2COC(=O)O2)=O)C(CNC(C2(C(F)F)CC2)=O)CC2COCC12 23121,C1(CC(=O)Nc2cccc(Oc3nccs3)c2)CCC2(CCCC2)CC1 23122,N1(C(c2cnc(C(C)C)s2)=O)CC(NC(C2CCS2(=O)=O)=O)CC(C)(C)C1 23123,N1(C(c2c(C)ccnn2)=O)C2CCCC1CN(C(c1cnc(O)cc1O)=O)C2 23124,CCS(=O)CC(=O)NCC1COCC1NC(=O)CSc1cn[nH]c1 23125,c1(CCC)c(C(N2CCCC(CNC(C3CCCN3CC)=O)C2)=O)nnn1CC 23126,C(=O)(C(CNC(c1cnsc1C)=O)CC(C)C)NC(c1c(C)nc(C)[nH]1)C 23127,Cc1cc(C(=O)NC(C)CCNC(=O)C=Cc2cnccc2C)ccc1C#N 23128,c1(-c2cnc3c(c2)N(C(C=CC=CC)=O)CC3)ccc2c(c1)n(C)c(=O)n2C 23129,c1(CNC(c2occc2CNC(C2C=CCCC2)=O)=O)ccc2n[nH]cc2c1 23130,c1(C(=O)NC(C)CCNC(=O)C(C)C2CCC2)ncccc1C(F)F 23131,n1(-c2cc(C)on2)c(C)cc(C(=O)NCC(C)NC(=O)C(F)C(C)C)c1C 23132,C1(CNC(=O)NC(C)CN2CCOCC2)CCCS1(=O)=O 23133,c1(N(C)Cc2nccc(C)c2)nc(=NC2CCN(C)C2)[nH]c2cc[nH]c12 23134,CC(O)C(C)(C)C(=O)NCC1CN(C(C2(CO)CCCC2)=O)CC12CC2 23135,C1(CNC(COCC#C)=O)CC2CCC(C1)N2C(C1CCCSC1C)=O 23136,c1(CC)[nH]c(=N)sc1C(N1CC(CN(C(=O)C=CBr)C2CC2)CC1C)=O 23137,C(=O)(C#CC1CCCCO1)NCCN(C(C(CSC)C)=O)C 23138,C1(C(C)CNC(C2CCC(=O)C2)=O)CCN(C(=O)Cc2cccc(Cl)c2)CC1 23139,C#CC1(O)CC(C(=O)N(C2CCN(C(=O)CCc3ccc(C)s3)CC2)CCO)C1 23140,CCC(CCOC)C(=O)NC12CCC(C1)N(C(c1sccc1-n1ccnn1)=O)C2 23141,CC1CN(C(C2CC3C=CC2C3)=O)CC1NC(c1cnn(C)c1N)=O 23142,N1(c2c(S(=O)(=O)NC3CCOC4(CCC4)C3)cccn2)CCOCC2(CCCC2)C1 23143,N1(C(c2ncc(C)c(C)c2)=O)CC(NC(=O)CC2CCCCN2C)C2(CCC2)C1 23144,N1(C(c2cn(C(C)(C)C)nn2)=O)CC2(NC(=O)C(c3ccc(F)cc3)F)CC1C2 23145,C1(N(C(c2c(C)ocn2)=O)C)CCCC(N(C)C(c2ccon2)=O)C1 23146,C1(C(c2ncc(C)o2)NC(c2nnnn2C2CC2)C)CCCCCC1 23147,Cc1cccc(C(N2CCOCC2CCNC(=O)CC2CCC23CCC3)=O)c1F 23148,C1(NC(C(C2CCCCC2)NC(c2ccc(CC)s2)=O)=O)CC2(CCC2)C1OC 23149,Cc1onc(Cl)c1NC(=O)C(=O)NCc1nccn1C(C)(C)C 23150,C1(NC(COC(C)C)=O)C2CC1N(C(c1ccnc(CN(C)C)c1)=O)C2 23151,N1(C(Cc2nc(NC(Cc3c(C)nn(C)c3C)=O)sc2)=O)CC2CCC(C1)N2C 23152,C1(CC(NOCC2CC(=C)C2)=O)CN(C(=O)C(C)O)CC1C 23153,C1(Cn2cc(C(C=C)(C)O)nn2)CCCN(C(=O)C(C)(C)c2ccc(Cl)s2)C1 23154,C1(C(=O)NCC2C(C)CCN2C(=O)Cc2cnco2)CC2CC1C1CC21 23155,C1(CC)CN(C(c2sccc2Cl)=O)CCN1C(=O)Cc1ccc(Cl)nc1 23156,c1(C(N2CC(CNC(C(c3c(C)cncc3)C)=O)C2)=O)cc2c(s1)CCSC2 23157,c1(CC(N2CCCC(NC(C3C(C=C)C3)=O)CCC2)=O)ccc2c(c1)CCCO2 23158,c1(C(C(=O)N(C(CNC(Cc2c(OC)cccc2)=O)C)C)C)cc(C)cc(F)c1 23159,c1(C(=O)NCCCCCN(C(CC2CCC(C)O2)=O)C)ccc(Cl)c(F)c1N 23160,C1(CC)C(NC(=O)C=C2CCC(C)C2)CCN1C(c1oc(C(F)(F)F)nc1C)=O 23161,C1(CC)(NC(=O)CCOCC2CCCO2)CCN(C(=O)C(C)n2cccc2)CC1 23162,c1(NC(c2c(COCC)nn(CC(F)(F)F)c2)=O)ccc2nn(C(C)C)cc2c1 23163,Cc1cc(C(=O)N(C)CCNC(=O)C(c2c(C)cccc2C)O)cc(C(F)F)c1 23164,C(C(=O)N1CCC(CO)(NC(=O)Cn2nnc(C3CC3)n2)C1)(C(C)C)OCC 23165,C(C(C)(CCO)NC(C1CCC2(CC2)C1)c1nnnn1C1CC(F)(F)C1)OC 23166,CC(C)CCC(O)C(=O)NC1CCN(C(=O)CC2(O)CCCCC2)CC1F 23167,N1(C(C2N(CC)CC2)=O)CC=C(C(C)(C)C(=O)NCCCOCC(F)F)C1 23168,c1(C(N2CC(C)(CNC(C(C3CC3)OC)=O)C2)=O)cc2c(cc1Br)OCCO2 23169,c1(CN2C(C(=O)NCC3(C)CC3)CSCC2)cc(I)ccc1O 23170,c1(C(=O)NC23CC2CCN3)ccc(S)nc1 23171,C(=O)(C1CSc2ccccc21)NCCC1CC(NC(c2c(CC)nn(C)c2)=O)C1 23172,N1(C(C(c2cnn(C)c2)C)=O)CCOC(C(=O)NC2COCC2CN(C)C)C1 23173,C(=O)(C(F)(F)CC(C)C)NC1CC2(C(NC(c3c(C)n(C)nn3)=O)C2)C1 23174,C1(C2CC2)(NC(c2c(C)cc(CC)o2)=O)CCN(C(C2CCCNS2(=O)=O)=O)C1 23175,CC1(NC(C2(NC(=O)CCc3ccccc3)CC(F)C2)=O)CCCC1O 23176,c1(CC2OCCN(OC(C=Cc3c(C)cncc3)=O)C2)c(Cl)cccc1[N+](=O)[O-] 23177,c1(N(CC(=C)C)C)nc(=NCC(C(C)C)N2CCOCC2)[nH]c2c1COCC2 23178,C1(CNC(c2ncncc2Cl)=O)CCCCN1C(=O)Cc1cccc(Br)c1 23179,c1(C(N2C(C(c3n(CCOC)nnn3)OC)C(C)CC2)=O)cnn(CCO)c1N 23180,c1(N(CCOCCN(C(c2ccc(SC)cc2)=O)C)C)cc(Cl)nc(SC)n1 23181,C1(NC(c2cc(OCC)ncc2)=O)CN(C(=O)C(O)CC(N)=O)CC1(C)C 23182,N1(C(c2ccc(Br)cn2)=O)CC2CCC1C1CN(C(C3(O)CCC3)=O)CC21 23183,c1(C(=O)NCC2CCCN(C(C3(O)C(C)(C)C3)=O)CC2)nc2ccccn2c1F 23184,c1(C(N(CC(CNC(C2C(C)OCCC2)=O)(C)C)C)=O)nccc2cccnc12 23185,C(CNC(=O)C=Cc1ncc[nH]1)(CCCC)NC(C1(CC#C)CCCO1)=O 23186,C1(CC(=O)N(C(c2ccccc2)C)CC2CC2)CCNCC1C1CC1 23187,CC1=C(C(=O)N2CCN(C(C3CC4C=CC3C4)=O)C(CCO)C2)CCS1(=O)=O 23188,C#CCCCCCCC(=O)NC1CN(C(C2COCCN2C)=O)CCC12CCC2 23189,CCCC(CC(C)C)C(=O)N1CCC(N(C(c2nocc2Br)=O)CC)CC1 23190,N1(C(c2ccc(C(=O)OC)o2)=O)CC(NC(=O)CCc2csc(C)n2)C(F)C1 23191,CC1=C(C)C(OC(c2cnc(C3CC3)nc2)=O)CCC1 23192,c1(NC(C(C)F)C)[nH]c(=NCCC(C)(C)S(C)(=O)=O)nc2c1ncn2C 23193,C12(C(N3CCC(N(C(c4c(C)cc(SC)o4)=O)C)C3)=O)CCC(CC1)C2(C)C 23194,C1(C2CCCO2)(C(=O)NCC(C(=O)OCC)C)CCCCC1 23195,c1(CNC(C(CSCC)n2cc(NC(C3CCC3)=O)nn2)=O)c(C)[nH]c(C)c1C 23196,c1(SCC)ccc(C(N2CCCC(CCNC(c3ccc(Cl)nn3)=O)C2)=O)cc1 23197,C(=O)(C1=NOC(C2(O)COC2)C1)NC(C)(CNC(c1ccc(C(F)F)s1)=O)CO 23198,N1(C(C2=CC(C)C2)=O)CCN(C(c2coc3ccccc23)=O)CC(O)C1 23199,c1(OC)c(C(c2nnnn2C)NC(C)CCC(=O)OC(C)COC)cccc1F 23200,Cc1ccc([N+](=O)[O-])c(C(=O)NC(CNC(=O)C(C)CF)CC(C)C)c1C 23201,C1(NC(C=C2CCC(C)C2)=O)CN(C(c2nc(=O)n(C)[nH]2)=O)CC1CC1CC1 23202,C1(C)(NC(c2cc(OC)ncc2)=O)CCCN(C(=O)CCc2cncc(O)c2)C1 23203,C1(CNC(c2c(Cl)nc(OC)s2)=O)CCCCN(C(=O)C(C)C2CC2)CC1 23204,C1(CC(=O)N(C)CC2N(C(C3(C#C)CC3)=O)CCC2)CCCC(=O)N1 23205,CCC(C)C(C(=O)NC(C)CNC(c1cccc(NC(N)=O)c1)=O)NC(=O)OC 23206,C(C(F)(F)CCC(=O)NC(C)CCc1ccc(C)cc1)n1cc(CCOC)nn1 23207,c1(C(=O)NC2(CNC(C3(OC)CCOCC3)=O)CCOC2)cc2ncccc2o1 23208,C(=O)(CCC#Cc1ccccc1)NC(C)CCNC(c1ccn2ncnc2c1)=O 23209,C1(CNC(CC2CC(C)(C)C2)=O)CCCCN(C(=O)CC2CCCO2)CC1 23210,C1(C(=O)NCC(O)CN(C)C(c2sccc2CC#N)=O)(COC)CC=CCC1 23211,CC1Oc2c(C(=O)NC3(CCNC(c4cccs4)=O)CC3)cccc2NC1=O 23212,N1(C(c2csc(C)c2C)=O)CC2CCC(NC(C3SCCS3)=O)(C2)C1 23213,Cc1c(C(=O)NCC(F)CNC(=O)CC2(C(F)(F)F)CC2)cccc1O 23214,N1(c2c(C)nccn2)CCC(O)C(C(=O)NCC2CCCC(=O)N2C)C1 23215,C#Cc1ccc(NC(=O)C(CNC(=O)C(C)C(C)CC)CCC)cn1 23216,N1(CC(=O)NCCCCc2ccc3c(c2)OCO3)CC(=O)NCCNC(=O)C1 23217,C(=O)(C(O)CNC(=O)CCC1CCCCC1)N1CC(CCOC)C1 23218,N1(C(C2(c3c(C)ncs3)CC2)=O)CC2(CCN2C(=O)CCCCNC(N)=O)C1 23219,CCCCC(O)CCC(=O)NC(CNC(c1ccc2nc(S)[nH]c2c1)=O)C(C)C 23220,C1(C(=O)NC2(C)CN(C(C3CCCN(C(C)=O)C3)=O)C2)CC2CC1CC2(F)F 23221,N(C1CCc2c(Br)cccc21)C(C1CC1C(=O)Nc1cccc2nc(O)oc12)=O 23222,C1(NC(Cc2cc(OC)cc(OC)c2)=O)Cc2ccccc2N(C(=O)C(C)O)C1 23223,c1(CNC(Cn2ncc(CC)c2)=O)cccc(C(=O)NCc2[nH]nnc2C)c1 23224,C1(C(N(CCCN2CCNCC2)C)=O)CC2(CCO1)CC(F)(F)C2 23225,c1(CNC(c2ccncc2CO)c2n(CCC3(C)CC3)nnn2)ccc(F)cc1 23226,c1(OCCC(=O)NCC2CCCN2C(c2nn[nH]c2Cl)=O)ccccc1F 23227,CC1CCCC(C(=O)NCCC2CCN(C(C3CC4CC3C4)=O)CC2)C1 23228,N1(C(=O)NCCc2ccon2)CCC2(CC1)CC2c1cccnc1 23229,Cc1ncnc(C(=O)NCCC2CCC(NC(=O)CN3CCNC(=O)C3)C2)c1C 23230,C1(NC(c2cnn(CC)n2)=O)CCC2(CC1)CC2NC(=O)CCC1CCCCO1 23231,c1(CC(=O)NC(C)C(CO)NC(c2nn(C)cc2N)=O)cnc2cccnn12 23232,S(=O)(=O)(c1c(C)sc(C)c1Br)NCc1c(OC(C)C)ccc(OC)c1 23233,C1(COC)CCCCN1C(C1CC2CC2N1C(C1CCCCCC1)=O)=O 23234,N1(CC)CCC(NC(=O)C(C)(C)CNC(C2CC=CCO2)=O)C(C)C1 23235,O=C1CCc2cc(-c3ccnc(C(=O)NCCc4ccc(O)cc4)c3)ccc2N1 23236,O=C(C1=CCCCCC1)NCC12CCC1CN(C(c1nncs1)=O)C2 23237,CC(CC(=O)NCC1(F)CCN(C(c2cnc(Cl)cc2N)=O)C1)C(C)(C)C 23238,C1(NC(c2c(NC(c3c(C)nsc3)=O)ccs2)=O)CC(O)C(O)C1 23239,c1(C(=O)OC)cnn2c1CC(Nc1nn3cc(CC(C)C)nc3s1)CC2 23240,C(=O)(C(CC)CCCCC)N1CC2C(NC(CCC=CC)=O)(C2)C1 23241,Cc1c(N2CCCC(CNC(=O)CCc3nc[nH]n3)CC2)ncnc1Cl 23242,C12(NC(c3ccc(CC)c(C)c3)=O)CCCC1N(C(c1cncn1C)=O)CC2 23243,c1(C(N2C(CNC(C(N3CCC(O)CC3)C)=O)CCC2)=O)cnn2ncccc12 23244,C(=O)(C1Cc2ccc(F)cc21)N1CC2(CN(C(CS(CC(=O)OC)(=O)=O)=O)C2)C1 23245,N1(C(=O)NCCOCCC(=O)O)C=CCCCC1 23246,Cc1cc(NC(=O)NCC2(Sc3ccccc3)CCCCC2)cnc1Br 23247,C12(NC(Cc3c(C)ocn3)=O)CCCN(C(c3ccc(Cl)c(F)c3F)=O)CC1C2 23248,C(=O)(C1=NOC(C(C)(C)C)C1)N1CCCC(N(C(C2C3CCC(F)C23)=O)CC)C1 23249,N1(C(C(COCC)n2cc(C3CCCC4CC34)nn2)=O)CCN(C)C(C(F)F)C1 23250,c1(CNC(=O)OC(C)(C)C)c(Br)sc2nnsc12.C(C1C(=O)N1)OC.C12CC1C2 23251,C(=O)(C1=CC2C=CC1C2)NC1(C2N(C(C3=CCCC3C)=O)CCCC2)CC1 23252,C(F)(c1ccccc1)=CC(=O)NC(CNC(C(COC)OC)=O)CC(C)C 23253,Cc1ncncc1C(=O)N(CC(C)N(C)C(C1CCCN(C)C1)=O)C 23254,C1(C(=O)NC(CN2CCN(C(C(=O)NCC)C)CC2)(C)C)CC2CCC1CC2 23255,c1(CCNC(CN2CCCC(CNC(CC)=O)C2)=O)ccc2cnccc2c1 23256,C1(C(NOCCCC)=O)CC(O)CN1C(c1ccn(CC)c1C)=O 23257,Cc1ccc2c(c1)C(NC(C1CN(C(c3ccsn3)=O)CCO1)=O)CCCN2 23258,N1(C(c2ccc(C(C)(F)F)cc2)C(=O)NC2CC2)CC=C(c2ccccn2)CC1 23259,C(CN=c1cc(C)nc(-c2cccc(Cl)c2)[nH]1)NC(C1CCC(OC)C1)=O 23260,c1(CC(=O)NCC(Cn2cc(C3(C)CCCO3)nn2)OC)c(F)cccc1Br 23261,N1(C(CC(C)C)=O)C(CNC(=O)Nc2cnccc2C(C)(C)C)CC2CC12 23262,CC(C)C(C(=O)N1CCN(C)CC1)C(C)NC(c1ccc(O)nc1)=O 23263,C(=O)(C(F)CC(C)(C)Nc1ccc(C)cc1)N(C(=O)CC1CC2CCC1C2)CC 23264,c1(NC)ccc([N+](=O)[O-])cc1C(N1CCC2(CCCN2C(=O)C=CCF)C1)=O 23265,C(C1COCc2ccccc21)NC(=O)NC1CCCC(C)(C)O1 23266,C1(NC(=O)NCC(C=C)O)CC(=O)N(c2ccccc2)C1.C1(=O)CCO1 23267,CC1ON=C(C(=O)N2CC(NC(=O)Cc3c(Cl)cnn3C)C(C3CC3)C2)C1C 23268,c1(OCOC)ccc(F)c(F)c1-c1ccc(CNC(c2ccc(F)cn2)=O)nc1 23269,N1(CC)CC(C)N(c2nc(C)nc(-n3cccn3)c2C)CC1C 23270,C1(NC(C)=O)CCC(C(N2CCC(NC(c3cn(C(C)C)cc3C)=O)C2C)=O)CC1 23271,N1(C(c2c(C)n[nH]c2)=O)CC2CC1(CNC(=O)C(C)(O)Cc1ccccc1)C2 23272,c1(C(N2CC(C(C)NC(c3c[nH]cc3-c3ccccc3)=O)C2)=O)nnc(S)n1C 23273,N1(C(C=CC=CC)=O)CCc2ccccc2C1CNC(=O)CCc1scnc1C 23274,N1(C(c2cncc(C(C)(C)C)c2)=O)CCN(C(c2csc(Cl)c2Cl)=O)C(CO)C1 23275,c1(-c2cc(NC(C3CC3(F)F)=O)sc2)ccccc1-c1ccco1 23276,c1(NC(C(CC)(C)CNC(=O)C(C)CN(C)C)=O)cnc2ccnn2c1 23277,C(=O)(C1=CC2CCCC12)NCC1N(C(c2cccc(C(C)C)c2N)=O)CCCC1 23278,N1(C(C(CC(C)C)C(C)C)=O)CCCC2(CCCN2C(=O)COCP(C)(C)=O)C1 23279,N1(C(C2(CNC(C(C)=NOCC#N)=O)CCCO2)=O)CC[Si](C)(C)CC1 23280,c1(C(=O)NCCCCOCC)c(-c2cncc(OC)c2)ncn1C 23281,Cc1cccc(CC(=O)NCCC(O)CNC(=O)CC2CC2)c1C 23282,CC1=C(C(=O)NCC2CCCN(C(=O)CCCc3nccs3)C2)CCC(C)(C)C1 23283,c1(C(=O)NCC2CCC(NC(C=CC=CCC)=O)C2)ccc(P(C)(C)=O)s1 23284,C1(CCCCNC(C(C)OC)=O)CCN(C(=O)CSc2nncn2C)CC1 23285,S(=O)(=O)(c1ccc(C#N)c(NC(CC)CCOCC)c1)NC1(C=C)CCOCC1 23286,N1(C(C=Cc2ccc(C)o2)=O)CC2CC(NC(=O)CCNC(=O)C=CCl)C1C2 23287,c1(COCC(=O)NC(C2CN(C(CCSCC)=O)C2)C)cc(C)no1 23288,Cn1nc(C(N2CCC(Nc3ncccc3C(F)(F)F)C2)=O)c2c1CCCC2 23289,c1(N2CCC(NC(c3nc(Cl)ccc3F)=O)(CF)C2)ncc([N+](=O)[O-])cc1Br 23290,C(=O)(C1=C(C#N)CCC1)N(C(C)C(=O)NC1CC(N2CCC2)C1)C1CC1 23291,N1(C(COCCSC)=O)CCC2(NC(C3CCN(C)C(=O)C3)=O)CCCCCC12 23292,C1(C(N(CC(CC)NC(=O)CC2COC(=O)C2)C)=O)CC2(CCC(F)(F)CC2)C1 23293,N1(C(CC(CCC)NC(c2oc(C)nc2CC)=O)=O)CCC2(CCCCC2)C1 23294,CCC(CC(F)(F)F)C(=O)N1CC2(CNC(C3CCC(C)CC3)=O)CC1CO2 23295,c1(C(=O)NCCN(C(=O)CC2CCCC23CC3)C(C)C)ccc(C(F)(F)F)cn1 23296,c1(C(=O)NCC(CN(C(c2ccsc2Cl)=O)CC)(C)C)cc2sc(C)cc2[nH]1 23297,N1(C(CCCC(=O)N(C)C)=O)CC2CCC1CN2C(c1ncccc1Cl)=O 23298,CC1(C)CCC(CNC(C2(C)CCCS2(=O)=O)=O)N(c2nnc(C3CC3)s2)C1 23299,N1(C(c2nc(C(C)C)oc2)=O)CCn2nc(C(=O)N(c3ccccn3)C)cc2C1 23300,c1(C(=O)NC(C2CC2C(=O)Nc2cncc(Cl)c2)C)ccnc(O)c1 23301,O=C(C1CCCn2c(Br)cnc21)NC12CC(C1)N(C(C1CC1F)=O)C2 23302,C1(C(=O)NC2(C)CCN(C(c3n(CC)cc(Cl)c3)=O)C2)CCc2ncnn2C1 23303,C(C(=O)N=S(C)(=O)c1cnn(C)c1CN)c1c(OCC(C)C)c2c([nH]1)cccc2 23304,C#CCCCC(=O)NC1CCOC(C2CCN(C(=O)Cn3ccsc3=N)CC2)C1 23305,CCS(=O)(=O)CC(=O)N1CCC(N(C(c2ccncc2)=O)C)C1.C1(N(C)CC)CC1 23306,N1(C(c2c(CNC(C3CCCN(C)C3)=O)c[nH]n2)=O)CC2C3CCC(O3)C2C1 23307,c1(C(=O)NC2C(NC(C3(C)CC4CC4C3)=O)CCOC2)cc2nn[nH]c2cc1F 23308,Cc1nnc2n1CC(C(=O)NC1CC1NC(=O)CCc1cc(Cl)no1)C2 23309,c1(C(CNC(C)=O)NC(C2N(C(c3cnsc3C)=O)CCC2)=O)ccc(F)cc1 23310,C1(CN(C(=O)CC2C=CCC2)C)COCCN1C(=O)Cn1cnnc1O 23311,N1(C(C2(C#C)CC2)=O)CCC(C(=O)Nc2cnccc2C)C(C)(C)C1 23312,C(=O)(C(O)CC(N)=O)N(CCCNC(=O)C=C1CCN(C)C1)CC 23313,C(=O)(CCC(C)NC(C1CC2(CC2)C1)=O)N(CC(O)CO)C(C)C 23314,Cc1cc(C(=O)NCC2CCC2NC(C2(CF)CCC2)=O)sc1Br 23315,c1(N2CC(O)(CNC(c3nn(C(CC)CC)c(C)c3)=O)C2)cc(O)nc(=O)n1C 23316,N1(C(C(c2ccc(C)o2)C)=O)CC(NC(c2onc(C)c2C)=O)CC(F)C1 23317,C1(CC)(CO)CCCN(C(=O)CC2COCCN2C(c2cn(C(C)C)cn2)=O)C1 23318,CC(C)CCC(C(=O)NCCCc1ncn(C)n1)NC(C1CC1(F)Cl)=O 23319,N1(C(CC(CC(C)C)C)=O)CCN(C(C2CC3CCC2C3)=O)CC2(C)CCCC12 23320,C1(NC(c2cccc(C(=O)NC)n2)=O)CN(C(c2noc(C)n2)C)CC1(C)C 23321,C1(C(N2CC(CCCCC)C2)=O)CCN(C(=O)C(C)CCOC)CC1C 23322,N1(C(=O)CC2CC2(Cl)Cl)CCC(O)(C(F)(F)F)CC1 23323,CC1CCN2N=C(C(=O)NC(C3CN(C(c4ccnn4C(F)F)=O)C3)C)NC2=N1 23324,N1(C(=O)OC(C)(C)C)CC(CNCC2CC(C)(C)CO2)C(F)C1 23325,c1(C(N2CC(N(C)C(c3n[nH]cc3F)=O)C2)=O)cn2c(Br)cnc2s1 23326,N1(C(C(CC)OC)=O)CCCC(C)(CNC(=O)CCc2cnco2)C1 23327,N(C1CCCc2ccc(F)cc21)C(C(CC)OC1CCCCC1)=O 23328,c1(NCc2[nH]nc(CSC)n2)nccc(=NCc2ccnc(C#N)c2)[nH]1 23329,CC1OC2(C(=O)OCC3CC(C#N)(Oc4ccccc4)C3)CCC1CC2 23330,C(C1CN(C(=O)CC(C)O)Cc2ccccc21)NC(Cc1ccn(C(C)C)n1)=O 23331,N#CC1CN(C(=O)C=Cc2ccc(O)cc2Cl)CCN1C(=O)C=Cc1ccsc1 23332,C1(CC)CN(C(C2CC(O)C(F)C2)=O)CC1C(=O)N(CC(N1CCCC1)=O)C 23333,C1(CNC(Cc2cc(C)n(C)n2)=O)CC12CCN(C(=O)C(C)(O)CC(F)F)CC2 23334,N1(C(c2ccnc(Br)c2F)C(=O)NCCSC)CC(CO)OCC12CCOCC2 23335,C(=O)(C1=CS(=O)(=O)CCC1)NC1C2(CN(C(c3cn(CC=C)nn3)=O)C2)CCC1 23336,C1(NC(C(C)CCO)=O)COC2(C1)CN(C(=O)Cn1nc3c(n1)CCCC3)C2 23337,CC1(C)NC(=O)CC1C(N1CC2C(CNC(=O)CC3CC4CCC3CC4)C2C1)=O 23338,c1(OC(C(=O)NC)C)ccc(NC(=O)Cc2sc(Br)nc2C)c(NS(C)(=O)=O)c1 23339,C1(F)(C(N(CC(C)N(C(C(c2cc(F)cc(F)c2)C)=O)C)C)=O)CCN(C)CC1 23340,N1(C(CCOCC)=O)CC2CCC1C2NC(c1nn(CC)cc1Br)=O 23341,N1(CCN(C)CC2CCCN2C(c2conc2C(F)(F)F)=O)C(=O)CNC1=O 23342,Cc1nccc(C(=O)NCCC2(C(=O)N(C3(CCO)CC3)C)CC2)c1N 23343,C#CCCCCC(=O)NC1(CN(C(=O)C=Cc2cc(Br)cs2)C)CC1 23344,C(=O)(C(F)C(=O)N1CC(F)CC1C(=O)N(CCCN=[N+]=[N-])C)OCC 23345,CC1CN(C(=O)C=Cc2ccco2)CC2(CCN(C(C3CCC(C)(C)O3)=O)C2)O1 23346,O=C(CS(=O)(=O)c1ccncc1)N(C1CCCC1)CC(=O)O 23347,O=C(N=c1[nH]nc2n1CCCC2)N1CCC(Cc2cccnc2)C1 23348,CCCS(=O)(=O)CC(=O)N1CCN(C(=O)CCOc2ccccc2F)C2CC12 23349,Cc1cc(=NCc2cccc(CN(C)C)c2)[nH]c(N2CCc3ncn(C)c3C2)n1 23350,c1(C(=O)NCCc2ccc(C(N(C)C)=O)cc2)c(F)ccc2n[nH]cc12 23351,N1(C(C2(C#C)CCC2)=O)CCC(C2CCCN(C(=O)C(C)C(C)(C)C)C2)CC1 23352,N1(C(CC(CCC)C)=O)CC2CCC(N(C)C(c3ncc(F)cc3C)=O)C2C1 23353,N=C1NC(=O)C(CC(=O)NCC2(O)CN(C(c3cc(C(F)F)no3)=O)C2)S1 23354,C1(CNC(c2c(CC)ncs2)=O)C(O)C(O)CN1C(=O)CN1CCCC1=O 23355,CC12CC(C(=O)NC3CC(O)CN(C(c4cnc(C(F)F)s4)=O)C3)(C1)C(C)(C)O2 23356,C(=O)(C#CC1CCOCC1)NC(C1CCCN1C(c1cc(C(F)(F)F)n[nH]1)=O)C 23357,C1(C)(C(=O)NCCN(C(CC=CC=C)=O)Cc2ccccc2)CC(OC)CN1C 23358,c1(CC(N2CC(NC(C3CC(C)(C)C3)=O)C3(C2)CC3)=O)ncn2c1COCC2 23359,C1(NC(CCOc2ccc(C)c(C)c2)=O)CC2(CCN(C(=O)CCC(C)O)C2)C1 23360,c1(C(N(CC(C)NC(C(CSC)C)=O)C)=O)cc2ccc(Cl)cc2c(O)n1 23361,N1(C(C(c2ccc(C)cn2)(F)F)=O)CCCC(NC(c2cccs2)=O)C1C 23362,C1(CNC(c2c(C)[nH]cc2)=O)CN2CCCCC2CN1C(c1ccn(C)n1)=O 23363,c1(C(N2CC(NC(CCOc3cccc(C)c3)=O)C(C)C2)=O)cc(O)nc(Cl)c1 23364,c1(C(=O)NC2CCN(C(C3CNC(=O)N3)=O)CC2F)cc2n(n1)CCNC2=O 23365,N1(C(C(=O)NC2COC2)C2C(C)C2)CCCC(C2CCC2)C1 23366,c1(C(=O)NCC2(F)CC(NC(C3CCSC3)=O)C2)cccc(CC(F)(F)F)c1 23367,CC1=NNC(=O)C1CC(=O)NCC1(CN(C)C(c2ccn(CC(C)C)n2)=O)CC1 23368,CCCC(CNC(=O)CC1CCN(C(=O)CC2(COC)CC2)C1(C)C)CCO 23369,C(=O)(CS(=O)(=O)CC(C)C)NC1(CCNC(c2ccnc(C)n2)=O)CC1 23370,C1(CNC(c2ncn(C)n2)=O)CN(C(=O)Cc2n[nH]c(=N)s2)C(C)(C)C1 23371,CC1CCCN1CCn1cc(CCC2CCCCC2)nn1 23372,C=CC1(CC(N2CCC2C(=O)OC)=O)CN(C(=O)C(COC)CC)C1 23373,N(C(=NCCc1csc(C)n1)NC1CC(c2ccccc2Br)C1)C(C=C)C 23374,n1(CC)cc2ccc(C(=O)N(C)CCNC(=O)CNC(C3CC3C)=O)cc2n1 23375,c1(N2CC(C(C)NC(C3(C)CCC(=O)N3)=O)C2)nc(Cl)nc2[nH]c(O)nc12 23376,C1(C(N2CCC(CCCO)C2)=O)CC2CC2N1C(=O)C(O)c1ccsc1 23377,c1(C(N2CC(Cn3cc(-c4scc(C)n4)nn3)OCC2)=O)c(O)ncc2c1CCC2 23378,N1(C(C(CCSC)(C)C)=O)CC2ON=C(CNC(c3coc(C(F)F)n3)=O)C2C1 23379,c1(N2CC(NC)C3(C2)CC3)ncc(C)cc1S(=O)(=O)NCc1cc(Cl)nc(Cl)c1 23380,Cc1nscc1CC(=O)N(C1CCC(NC(=O)COC(C)C)C1)C 23381,c1(N2C(C)C(NC(=O)CC3(C)CC3)CCC2)ncc2ccnc-2[nH]1 23382,N1(C(C(N2CCN(C)CC2)C)=O)CC2CN(C(C3(Br)CC3)=O)CC(C1)O2 23383,c1(CSC)cccc(C(=O)NC2(C)CCN(C(c3nncs3)=O)C2)c1 23384,CC(C(O)C(F)F)NC(=O)C(c1ccco1)NC(=O)CC1(C)CCOC1 23385,C(C1=CCCSC1)(c1nnnn1C1CCOCC1)NCCCCC(C(C)C)O 23386,C1(OC)CCN(C(=O)C(CN)C2CCCCC2)CC1(C)C 23387,N1(C(COCCC(C)C)=O)CCC(C)(C)C1CNC(=O)CSc1cccnc1 23388,N1(C(COC)=O)CC2CCCC(NC(C3CCC=CCC3)=O)(C2)C1 23389,N1(C(C(CC=C)C(C)C)=O)CC2(CCN(C(c3cc(C)c[nH]3)=O)CC2)CC1C 23390,N1(C(C2C(OCC)C2)=O)CC2CCN(C(=O)CCc3cc(C)nn3C)CC2C1 23391,c1(C(N2C(C)CC(NC(c3coc(S(N)(=O)=O)c3)=O)C2)=O)cccc2c1OCC2 23392,C(CC(O)C(=O)N(Cc1ccccc1)OC)NC(C1N(CC)CCOC1)=O 23393,C1(NC(C(C=C)O)=O)CCCOC12CCN(C(c1ccc(C)c(F)n1)=O)CC2 23394,CC1(C)CC(CC(=O)NCC(CNC(=O)CCNC(=O)CO)CO)CCO1 23395,c1(OCCOC)ccc(Cl)cc1C(=O)NCC1CN(C(=O)C(C)CF)CCO1 23396,CC(C)C(C)CC(=O)N1CC(C)CCC1C(=O)Nc1cc(Cl)cnc1O 23397,c1(OC)nccc(Br)c1C(=O)N(CCCNC(C1CCSC1)=O)C 23398,N1(C(c2nc(C)oc2)=O)Cc2[nH][nH]c(=NC(=O)c3cc(Br)ccc3Cl)c2C1 23399,c1(C(N2CCC(OCCNC(CCC#CC)=O)C2)=O)cc(C)c(O)c(C)c1 23400,c1(SCC(=O)Oc2c(C(CC)=O)cccc2)[nH]c(=N)c(C#N)cc1C#N 23401,CCCCC(CNC(=O)CCSc1ccccc1)NC(=O)CCC1CCCN1C 23402,C(=O)(C1=NNC(=O)CC1)NC1CN(C(C2C(C)(C)OCC2)=O)CC(O)C1 23403,C1(O)(CC(=O)N(C)CC)CCN(C(=O)C(O)Cn2cncn2)CC1 23404,C1(C(=O)NC(C)CCNC(=O)C(C(C)O)N(C)C)(COC)CCCCO1 23405,CC1=C(C(=O)N2CCCC(NC(c3cc(F)ccc3Cl)=O)C2C)CCC1 23406,c1(NC)cccc(C(=O)NC(C)C(c2ccccc2)NC(=O)C(C)SC)n1 23407,c1(OCC#C)ncccc1C(=O)NCC1CC(NC(c2cnn(CC=C)c2)=O)C1 23408,S(=O)(=O)(c1cccc2c(Cl)cc(C)nc12)NCCN1CCC(NC)CC1 23409,C(C(CC1CCCC1)C(=O)NOCCN(C)C)NC(C1OCCC(C)C1)=O 23410,c1(C(N2CC3CN(C(C=CCN(C)CC)=O)CC3C2)=O)cc(F)c(F)c(O)c1F 23411,CC1(NC(=O)C(C2CCOCC2)O)CCCN(C(=O)CSCc2ccccc2)C1 23412,c1(C(=O)NCC2(O)CN(C(C(C)NC(CC)(C)C)=O)C2)cc(Br)cn1C 23413,CC1CCCCN1CCC(=O)N(CC(C)NC(=O)Cn1nnc(C(C)(C)C)n1)C 23414,c1(C(=O)NC2CN(C(CN(S(=O)(=O)Cc3ccccc3)C)=O)C2)cnc(O)[nH]1 23415,c1(OC)cccc(NCC2(NC(=O)CCNC(=O)OC)CCOCC2)c1[N+](=O)[O-] 23416,C=C1CC2(C1)CC(C(=O)NCC(C)CNC(=O)C(O)C(F)(F)F)C2 23417,C(=O)(CC(C1CC(F)(F)C1)NC(c1ncoc1C(F)F)=O)OCC 23418,c1(C(=O)OCCC(=O)Nc2ccc(OCC)cc2C)cnc2ccccn12 23419,N1(C(C(C(C)C)CNC(C2(C)CCC3CC3C2)=O)=O)CCCOC(C)(C)C1 23420,C1(CC)CCC(C)CN1C(c1c[nH]nc1CNC(c1cnc(Cl)s1)=O)=O 23421,C1(N(C(=O)CCC2CCOC2)C)CCCN(C(=O)C(C)(C)c2ccccn2)CC1 23422,C1(O)(CNC(c2c(C)csc2)=O)CCCN(C(c2cc(Cl)nnc2O)=O)C1 23423,N1(C(C2CCCN(CCC)C2)=O)CCC(NC(=O)CN2C(C)CCC2C)C(F)C1 23424,CC1CCN(C(=O)CCc2cncc(F)c2)C1CNC(=O)CSCC(F)(F)F 23425,c1(CC(=O)NC2(CNC(C(Br)=C(C)C)=O)CCC2)cc(C(F)(F)F)c(O)nn1 23426,c1(NC)cncc(C(=O)NC2COCC2CSc2ccccc2)c1 23427,C1(C(=O)NC(C(C)NC(C2CC3(CC(=C)C3)C2)=O)CO)CCC2(CCCC2)CC1 23428,N1(C(C(C)NC(COC)=O)=O)CC2CC1C2CNC(C1(C)CC1(F)F)=O 23429,c1(C(C)NC(c2ccc(C)nc2)c2nnnn2C2COC2)ccc2nc[nH]c2c1 23430,c1(C(N2CCN(C(C(n3ccc(C)n3)C)=O)CC2CF)=O)ccc(O)c(C)c1C 23431,C1(NC(C=COCC)=O)COCCC1NC(=O)C(O)CCc1ccccc1 23432,n1(CC=C)cc(C(=O)NCCCN(C(=O)CSCC2CCOC2)C(C)C)nn1 23433,C(=O)(C1=NOC2COCC12)N1C(C)CC(CC(N2CC3CCC=CC23)=O)C1 23434,CC1(C)C(CNC(C2(N3CCNC3=O)CC2)=O)CCN1C(=O)CCSC1CC1 23435,C1(CC2(O)CCN(C3CC(=O)N(CC)C3=O)CC2)COC2(CCCC2)O1 23436,C1(C(N(CCCC)CC)=O)CN(C(C2CCCOC2)=O)C(C)(C)C1 23437,C12(OC)CCC(C(N3CCC4C(NC(c5cc(C)cs5)=O)CC34)=O)(CC1)CC2 23438,c1(C(=O)NC2CC3CC(NC(C(C(C)(C)O)F)=O)C2C3)ccn2cccc2c1 23439,C(=O)(C(O)(C(C)C)C(F)(F)F)N1CCCCC(NC(c2c(C)scc2)=O)C1 23440,N1(C(=O)NC)CCN(C(=O)CC2CC2CNC(c2ncco2)=O)CC1 23441,c1(CNC(=O)CC2CC(=O)NC2=O)ccc(CNC(=O)COC2CCC2)c(F)c1 23442,C(=O)(C(CC(F)F)NC(=O)Nc1cc(C)cnn1)OCC 23443,N1(C(C(C)C)=O)CCN(C2CCC(NC(=O)C(N3CCC(C)(O)C3)=O)C2)CC1 23444,c1(C(C(=O)NC(CCOC)CNC(c2cc(C)sn2)=O)C)cccc([N+](=O)[O-])c1 23445,N1(C(c2ccc(C#N)cn2)=O)CCC(NC(=O)CCF)C12CCC2 23446,C1(NC(C2N(CCC(C)C)CCC2)=O)CN(C(=O)Cn2nccn2)CC1CO 23447,N1(C(C(C(C)O)C)=O)CCC(C2(NC(c3ccccc3)=O)CC2)C1 23448,C1(NC(C)(C)COC(c2ccco2)=O)CC2(C1)CC(C#N)C2 23449,C(=O)(CC(F)(F)C(F)F)N1CCC(NC(c2cc(COC)sc2)=O)C(F)C1 23450,C(=O)(C(O)(C(C)C)C(F)(F)F)NCC(C)NC(Cc1c(C)ccnc1)=O 23451,C1(C(C)NC(=O)C(O)C2CC2)CN(C(C2(C(N)=O)CC2)=O)C1 23452,CC1CC(NC(c2cccn2C)=O)CN1C(C1CC1C)=O 23453,C1(N(CC(=O)Oc2cccc(C)c2)C)CCC12CCN(C(=O)OC(C)(C)C)CC2 23454,c1(NC(C2CCCN2C(=O)CN2CCOC2=O)=O)cnc2ccccc2c1Cl 23455,Nc1cncc(C(=O)NCC2CCCCN2C(c2cc(C(F)(F)F)ccn2)=O)n1 23456,C1(C(=O)NCCN(C)C(c2ccc(-c3nccs3)cc2)=O)CS(=O)(=O)CC12CC2 23457,Cc1c[nH]c(C(N2CCCC2CNC(c2cc(Cl)ns2)=O)=O)c1 23458,C1(NC(COCc2onc(C)n2)=O)CN(C(C2CCN2C2CCCC2)=O)CC1F 23459,Cc1cc(C(N2CCN(C(c3ccc(Br)c(O)n3)=O)C3CC23)=O)nc(C)c1 23460,Cc1cnc2cccc(C(=O)NC(C)CCNC(C3CCCCO3)=O)c2c1 23461,N1(C(CSCC#C)=O)CCN(C(=O)Cc2cn3ccsc3n2)C(CO)C1 23462,c1(C(=O)NC2CN(C(C(c3cccc(C)c3)(C)C)=O)C2)ccc(F)c2[nH]ccc12 23463,c1(C(=O)NC(C)CC(N)=O)cccnc1CNC(c1nn(C)cc1Cl)=O 23464,C=CCC(C(=O)NC1CC1C(C)(C)C)NC(c1sccc1Cl)=O 23465,C1(CC(=O)NC(CCCNC(C2CC(OC)C2)=O)c2ccccc2)CCCCO1 23466,N1(C(c2c(CC)nns2)=O)CC(C)C(C)(CNC(c2nccnc2N)=O)C1 23467,c1(C(N2CCCC2(C)c2ccccc2)C(=O)NC)cccc(C(F)(F)F)n1 23468,N1(C(C2CC(OC)(OC)C2)=O)CCC(C)C(CC(=O)NC(c2nc(C)no2)C)C1 23469,N1(C(c2cnn(C)c(=O)c2)=O)CC(C(N2C3C=CCC2CC3)=O)CCC1(C)C 23470,CCCCC(C(=O)NC(C)CCCCNC(C)=O)N1CCCS1(=O)=O 23471,CC(F)(F)CCCC(=O)NC(CNC(C1OCC1(C)C)=O)CO 23472,C1(CSC)CCCN(C(=O)CCN(C(=O)C(F)=C2CCC2)C(C)C)C1 23473,C(=O)(CCCCCN(C)C)NC1C(CNC(C(C)COc2ccccc2)=O)C1 23474,NC(=O)CCC(=O)NCC1(C(=O)NCc2ccccc2F)CCCO1 23475,CC1(C)CCC(n2cc(CCNC(N)=O)nn2)CN1C(C1CC12CCOCC2)=O 23476,CC(C)CCCC(=O)N1CCCCC1CCN(C)C(c1cc(CC(C)C)c[nH]1)=O 23477,CC(C)(F)CCC(=O)NC1CCCC1CNC(c1cccc(Br)c1F)=O 23478,N#Cc1ccccc1C=CC(=O)NCC1(NC(c2n[nH]cc2F)=O)CCOC1 23479,Cc1cc(C#N)nc(N2CCC(N(C)C(c3ccn4ccnc4n3)=O)C2)n1 23480,C1(N(C(=O)C(C)NC(=O)C2CC2)CCC)CCN(C(=O)CCC(=O)OC)CC1 23481,CCC(CC(F)F)C(=O)NC1CCC1NC(=O)C(C(C)C)NC(=O)CCCOC 23482,C1(NC(C(C)=C2CC2)=O)CN(C(c2ccc([N+](=O)[O-])c(C)c2)=O)C2CCCCC12 23483,c1(C(=O)NC2C(NC(CCCC(C)C)=O)CCCC2)cc(F)cc2c1CCC2 23484,Cc1ccc(Cl)c(C(N2CC3(CCC3)CC2CNC(C2(CF)CC2)=O)=O)c1N 23485,c1(OC)cnc(Cl)cc1C(=O)NC1(CO)CN(C(C2CCCC(=O)N2C)=O)C1 23486,C(=O)(C(C)(C)c1sccc1Cl)N(CC(C)NC(=O)CCNC(=O)C=CCl)CC 23487,N1(C(c2ncn(CC)n2)=O)CCOCC(C(=O)NCC(C(C)C)N(C)C)C1 23488,c1(NC(COc2ccc(CNC3C(CC)CCC3)cc2)=O)nc(O)sc1C 23489,C1(NC(CN(C(=O)CC2CCCOC2)CCC)=O)CCN(C2CC2)C1=O 23490,c1(N2CC3N(C(C4(O)CC4)=O)C(CC3)CC2)nc2ccc(F)cc2s1 23491,C1(CNC(COC(CC)C)=O)CCCN(C(c2cn[nH]c2)=O)C1 23492,CC(CC#N)C(=O)N1CC(n2cc(C(C)N(C)C)nn2)C1 23493,C(=O)(CC1=CCN(C)CC1)NCCC(N1C(C)CS(=O)(=O)CC1)=O 23494,N1(C2(c3cn(C(C)C)nn3)CCC2)CCCN(C(c2ccc[nH]2)=O)CC1 23495,C1(CC(=O)NC2CC2(F)F)CN(Cc2ccc(-c3ncccn3)cc2)CCO1 23496,c1(CN(CCNC(C2CCCO2)=O)C(C2CC(OC(F)F)C2)=O)ccccc1 23497,C#CC1CN(C(=O)CC2CCCCN2C(=O)CC2CCC(=O)C2)CCN1C 23498,Cc1nc2cncc(C(=O)N(C3CCN(C(=O)C(C)(F)C(C)(C)F)C3)C)c2[nH]1 23499,C=CC(C)(C)C(=O)Nc1cccc(CNC(=O)C(c2ccnn2C)C)c1 23500,c1(OC)c(C)cc(C(=O)NC2CCCC(N(C(=O)CSC3CC3)C)C2)cc1C 23501,C1(CC#C)(C(=O)NCC2(O)CCOCC2)CCN(C(=O)CC2CCOC2(C)C)C1 23502,c1(CNC(C(C2CC(NC(C(C)SC)=O)C2)F)=O)cc(C)ccc1C 23503,N1(C(Cc2cn(CC)nc2)=O)C2CC1CN(C(C1CCCN1C(C)C)=O)C2 23504,c1(C(N(CCNC(C2C(COC)C2)=O)C)=O)cccc(Cl)c1O 23505,c1(C(=O)NCC2CCCN(C(c3ccon3)=O)CC2)c[nH]c2ccc(Br)cc12 23506,c1(COC)ccccc1CC(=O)NC(C)CNC(=O)Cc1cc(C)nn1C 23507,c1(C(=O)NCC(C)C)cccn(O)c1=O.C1(C)(C)C2(CC2)CO1 23508,c1(C(N2CC(SC)C(NC(=O)C(O)C(C)C)C2)=O)cc(S(N)(=O)=O)cnc1C 23509,N1(C(C(C(CC)C)OC)=O)C2CCC1CN(c1ncnc(Cl)c1OC)CC2 23510,C(=O)(C(O)C(C)SC)N(C(c1cccc(OC(c2cnc(OC)s2)=O)c1)=O)C1CC1 23511,C(=O)(CC1OCCc2ccsc21)N(CCCNC(C1CC2C(C1)C2(C)C)=O)C 23512,Cc1csc(C(C)CNC(=O)C=Cc2ncc[nH]2)n1 23513,c1(C(=O)O)ccccc1C.Cc1nc[nH]c1C(N1CCC1(C)C(=O)N)C1CC1 23514,N1(C(CSCCNC(Cc2n(C)nnc2)=O)=O)CC2CC2C2CC12 23515,n1(CC(=O)[N+](CCC2CCN(CCCC(=O)N(CC)CC)C2)([O-])NC)ncn(C)c1=O 23516,C(=O)(CCC(CF)CF)NCCn1ccc(C(N2CCC(N(C)CC)C2)=O)c1 23517,N1(C(COC)=O)CC2C3CCC(C2C1)N(C(c1occc1-c1ccccc1)=O)C3 23518,N1(C(C2C(OC)CCC2)=O)CCC2(CCN(C(=O)CN3CCCCC3)CC2)C1 23519,c1(C(C)C(N2CCCC2C2CCN(C(C3CN(C)C3)=O)C2)=O)ccc(F)cc1Cl 23520,Cc1cc(Cl)cc(C(N2CCCOC(CNC(C3CC4(CCC4)C3)=O)C2)=O)c1C 23521,c1(C(=O)NCCN(C(=O)CC23COC(C2)C3)CC)ccc(C(F)F)s1 23522,C1(C(N2CCC(NC(Cc3c(C)ccc(C)c3)=O)C2)=O)(CF)CCC(F)(F)CC1 23523,N1(C(C(C)(C)SC)=O)CC2CS(=O)(=O)CC2(NC(c2ccc3cccnn23)=O)C1 23524,N1(C(C(COC)O)=O)CCOCC(F)(CNC(=O)CCc2ccccn2)C1 23525,CCS(=O)(=O)CC(=O)N1CCN(C(=O)CC2C=CS(=O)(=O)C2)C(CO)C1 23526,c1(CC)ccc(C(=O)NCC2COCC2NC(c2c(C)cncc2C)=O)cc1Cl 23527,C(=O)(CC(F)(F)CC)N1CC(C(=O)NCC2N(CC)CCC2)C(O)C1 23528,C1(CC)CN(C(=O)CCC(F)F)CCC1NC(=O)Cc1nc(C2CC2)cs1 23529,C1(NC(c2c(C)nn(C(C)(C)C)c2)=O)CC2CCC1N(c1ncncc1C#N)C2 23530,C1(O)(C(=O)NCC(C)CNC(=O)C(n2ccc(C(F)(F)F)n2)C)CCCCCC1 23531,C1(CNC(C(C2(O)CCOCC2)(C)C)=O)CN(C(C2CSCCS2)=O)C(C)(C)C1 23532,c1(CNC(=O)NC2C(C(=O)OC)CNC2)ccc(O)cc1Cl 23533,CCCC(C(C)(C)C)NC(=O)CC(C)(C)NC(C1CCCN1C(C)=O)=O 23534,c1(CC)ccccc1OCC(N1CCCC1CNC(=O)C(C)(C)c1cnco1)=O 23535,CCCC(C(F)(F)F)NC(C1CCCC(NC(=O)C(C)=C2CC2)CC1)=O 23536,C1(OCCCNC(CC2CC(CC)C2)=O)CCN(C(=O)CC2CCOC2C)CC1 23537,c1(C(=O)NC(CNC(c2ccc(CCC)[nH]2)=O)CC)ccc(NC)cc1Cl 23538,N1(C(C(C(C)C)O)=O)CC2=C(C1)CN(C(c1cccnc1-c1nncn1C)=O)C2 23539,C1(CNC(CC)=O)CC(NC(c2ccc(=NC)[nH]c2)=O)C12CCC2 23540,c1(C(=O)NC2CCCC(NC(CC(C=C)C)=O)C2)n[nH]c2cccc(OC)c12 23541,Cc1cc(C(=O)N(CCC(C(C)C)NC(=O)CC2CCCO2)C)c(C)nc1C 23542,O=C(CC1CCc2ccccc21)NC1CC2CN(C(=O)CC3(CO)CCC3)CC12 23543,CC1CCN(C(=O)C(F)CC2CC2)CCN1C(=O)CC1NC(=O)NC1=O 23544,c1(C(=O)NC23CC(NC(C4C(C)(CC)C4)=O)(C2)C3)cc(F)cc(F)c1N 23545,CC(C)CS(=O)(=O)CC(=O)N1CC(NC(=O)CCc2cscn2)CC1(C)C 23546,Cc1cccc(C(F)CNC(C2CCCN(CC(=O)Nc3ccccc3)C2)=O)c1 23547,c1(C(c2n(CC=C)nnn2)NC2CCCC=C2Br)cn2cc(C)ccc2n1 23548,CC1CN(C(c2cccc(=O)n2C)=O)CC(C)C1NC(=O)Cc1cccs1 23549,C=C1COCCN(C(=O)CC(CC)N(C(=O)Cn2cnnn2)C)C1 23550,C(=O)(C#CC1CCOC1)N1C(CC)CN(C(c2cc(N)cnc2C)=O)CC1 23551,CCCC(C(=O)NC(CC)C(c1ccc(OCC)cc1)=O)N(C)C 23552,N1(C(=O)OC)CCCC(C(=O)N(CCNC(=O)C#CC(C)C)CC2CC2)C1 23553,c1(NCC(C2CCCCO2)(C)NC(=O)C)ncc(Cl)cn1.c1(C)ncoc1C1CC1 23554,C1(NC(=O)NCC(=O)Nc2c(CC#N)cccc2)CCCC(C)(C)C1 23555,c1(N(CCCCN(C(Cc2cnc(C)s2)=O)C)C)snc(Cl)c1C#N 23556,O=S(=O)(c1ccc(NCC2=CCCC2)cc1Br)NCc1cscc1Br 23557,N1(C(CN(C(=O)OC)C)=O)CCC2(COC(CNC(c3ccccc3)=O)C2)C1 23558,c1(CNC(C2(N(C(C3CC(C)OCC3)=O)C3CC3)CCC2)=O)cc(F)ccc1O 23559,c1(C(=O)NCC2(NC(C(C(CC)C)C)=O)CC(OC)C2)cc2cccnc2[nH]1 23560,CCCC(C)(C)C(=O)NCCC1(C)CCN(C(c2cn(C(C)C)nn2)=O)C1 23561,CN1CCCN(C(c2ccc(C#N)cc2F)C(=O)NCCC2CC2)CCC1 23562,C12CCCC(C1)NC(=O)CN2C(C1(N(C)C)CC1)=O.c1(CSC)ccccc1 23563,Cc1oc(Br)cc1C(N1CCC(O)C1c1cccc(Br)c1)=O 23564,C(C)(C(C(C)C)NC(c1ccc(C(F)(F)F)s1)=O)NC(c1ccn(CCC)n1)=O 23565,c1(N(C)Cc2cc(C)on2)nc(N2CC3CCC(CC3)C2)nc2ncn(C)c12 23566,S(=O)(=O)(c1cnc(NC2CC2C2CCC2)cc1C)NC(c1nc(C)cs1)CC 23567,c1(C(N(CC(=O)N(C(CN(C(C)=O)C)C)C)CC2CC2)=O)cn[nH]c1 23568,O=C(NNC(=O)c1cc(-c2ccc(Cl)cc2)[nH]n1)c1ccon1 23569,N1(C(C2N(CC)CC2)=O)CC(C2(NC(c3cccc(CO)c3)=O)CC2)C1 23570,c1(C(=O)Nc2ccc(C3(NC(COC)=O)CCC3)cn2)ccc2occc2c1 23571,c1(C(=O)NC(C(=O)N(C(C2CCCO2)C)C)C)cc(Cn2cnnn2)cnc1O 23572,N1(C(=O)Nc2cncnc2)CCC(c2nc(-c3ccc(Br)s3)no2)CC1 23573,N1(C(c2nncc(C)c2)=O)CC2CC(NC(=O)C(c3ccc(F)cc3F)C)C2C1 23574,C1(NC(c2cnc(-n3cccn3)cn2)=O)CCN(C(C2CC3CC3C2)=O)CC1O 23575,CC(N=c1[nH]c(=NCC(F)(F)Br)[nH]c2c1CSC2)c1cc(F)ccc1F 23576,CC(C)S(=O)(=O)CC(=O)N1CC2(CCN(C(c3ccn(O)c(=O)c3)=O)C2)C1 23577,c1(OC)cc(N(C)C)ccc1CNC(C1CC1C(=O)Nc1cncc(C)n1)=O 23578,N1(C(c2cnc(C)o2)=O)CC2CCCC2C1C(=O)NCCC1CC(F)C1 23579,C(CCSC)(C(=O)N(C)CC1(NC(=O)CC2CSCCS2)CC1)OC 23580,c1(C(=O)NCC2C(NC(C(OC)OC)=O)CCCC2)ccc2c(n1)CCC2 23581,c1(C(N2CCN(C(=O)CCN3CCCC3)C(C3CC3)C2)=O)ccn2nccc2n1 23582,CC1(C)C(C)(NC(c2sccc2CNC(=O)C(F)n2ccnc2)=O)C1(C)C 23583,C1(C(=O)NCC#CCOC)(CNC(C2CCC(C)(C)C2)=O)CC12CCC2 23584,C(=O)(C1=NOC(CNC(c2cccc(CO)c2)=O)C1)NC(C(=O)NCCC)C 23585,N1(C(CC2(COC)CC2)=O)CCCC(C)(C)C1CNC(c1ccc(C)c(F)c1)=O 23586,N1(C(C(CC#C)O)=O)CC2CCC(C1)N2C(=O)CC(C)(C)COC 23587,c1(C(N2C(C)CC(CNC(c3occc3Br)=O)C2)=O)cc2n(n1)CCC2 23588,C(=O)(C1=CCC(F)(F)CC1)N(CCCNC(C1(COC)CCCOC1)=O)C(C)C 23589,c1(C(=O)NC2CC(C)N(C(=O)C(C)(C)CCC#N)C2)ccc2nc(CO)[nH]c2c1 23590,C1(C(N2CCC(F)(CNC(c3nn(C)c(F)c3)=O)CC2)=O)CC2CCCCN2C1 23591,C(=O)(C(CCC(N)=O)n1cc(C2COCC2O)nn1)NC(c1cncs1)C 23592,Cc1ccc(CCC(=O)NC2CCCC2NC(C2(O)CCOC2)=O)c(Br)c1 23593,c1(C(=O)NC(C2CCOC2)C)ccc(-n2cccn2)cc1 23594,C1(OC(C)C(=O)NC(C2CCCN2C(C2CC(CF)C2)=O)(C)C)CCCCCC1 23595,C(=O)(C(C(=O)N1CCC(C(C)(C)NC(C2CCCC2C(C)C)=O)CC1)OC)OC 23596,N1(C(CCCOCCOCC)=O)CC2ON=C(CNC(c3cnn(C)c3)=O)C2C1 23597,C1(NC(C(n2cc(C)nc2)(C)C)=O)CN(C(c2ccoc2)=O)CCC1C(F)(F)F 23598,Cc1nn(C)c(C)c1-c1cn(C2CCCC2NC(C2CCC(=O)N(C)C2)=O)nn1 23599,C(=O)(C(CC(C)C)N(C(=O)CN1CC(=O)NC1=O)C)NCc1c(C)non1 23600,CCC(C)C(C)C(=O)NCCCN(C(=O)CCc1csc(C)n1)C 23601,N(C1CC(C)(C)Oc2ccc(F)cc21)C1CC(S(=O)(=O)N)C1.CCC 23602,n1(CC)cnc(C(=O)NCc2occc2C(=O)NC2(CC)CCC2)n1 23603,CCC(C)(C)C(=O)C(=O)N1CCCC1C(=O)NCc1noc(C(C)C)n1 23604,N1(C(CC(OCC)OCC)=O)CC(NC(c2ccc(Br)nc2Br)=O)C(C#N)C1 23605,S(=O)(=O)(c1c[nH]c(=NCCSc2ccccc2)cc1C)N1CC(C)=C(C)CC1 23606,CC(C)S(=O)(=O)CC(=O)N1CCCC(N(CCCOCC(F)F)C)C1 23607,C1(C(N2CCC(NC(CC=CC)=O)C23CC3)=O)CC(c2ccccc2F)=NO1 23608,N1(C(c2n[nH]cc2-c2ccccc2)=O)CCN2C(=O)OCC2C1 23609,Cc1cnccc1C(=O)NC1CC(CNC(=O)C(C)(C)n2cc(Cl)cn2)C1 23610,C1(C(N2CCC(CNC(C3CC(C#N)C3)=O)CC2)=O)CCC(=C(F)F)CC1 23611,c1(CC)ccc(N)c(C(N2CC3C(CNC(=O)CC4C(C)C4(F)F)C3C2)=O)c1 23612,N1(C(CC=CC=C)=O)CCN(C)CC1C(=O)NCC(C)C(F)F 23613,C1(C)(C(N2CC(C(C)NC(=O)C(c3ccccc3)F)C2)=O)CCCN1C 23614,N1(C(CNS(CC)(=O)=O)=O)CCC(NC(C2CCC(=O)N2C2CC2)=O)C1(C)C 23615,C(=O)(CC(C)(C)CC(=O)N1CCC1CNC(C1CCN(C2CCC2)C1)=O)OC 23616,c1(NC(C)=O)c(C(=O)NCC2C=CC(NC(=O)CN3CCCC3)C2)cccc1C 23617,C1(NC(=O)CCn2ccnn2)CCC(NC(=O)C(C2CC(F)(F)C2)O)C1 23618,C1(NC(C2CCS(=O)(=O)N2)=O)C2CC3CN(C(c4cnsn4)=O)C1C3C2 23619,c1(C(=O)O)cnn(CCC2CCN(CCC3CC3)C2)c1 23620,c1(NC(C2CC23CN(C(c2ccc(O)nc2)=O)C3)=O)cc2ccccn2n1 23621,Cc1ccc(C(=O)Nc2cnc(-c3ccccc3C)s2)c(N)c1 23622,N1(C(C2CCN(C(=O)OC)CC2)=O)CCC(C)(C)C1CNC(=O)C(C)N1CCC1 23623,CCCC(CC)CC(=O)NCC(O)CN(C)C(c1ccoc1CC)=O 23624,CC(c1cccs1)=CC(N1CCC(C(F)CNC(C23CC(C)C2C3)=O)CC1)=O 23625,N1(C(C(C)NC=O)=O)CCC(C(C)C(=O)NC2(c3ccsc3)CC2)C1 23626,N1(Cc2cnc(C)[nH]2)CCCC2(CCN(C(c3ncc(OCF)cn3)=O)C2)C1 23627,N1(C(c2c(F)ccc(F)c2Cl)C(=O)NCC(=C)C)CCc2[nH]nc(C(F)F)c2C1 23628,C#CCCC(C(=O)NCC1CCSCC1)NC(c1cc(CCC)[nH]n1)=O 23629,CCC(C)(COC)C(=O)NCc1ncoc1C1CN(C(C2CCN(C)C2=O)=O)C1 23630,N1(C(CC(C)N(C)C)=O)CCCC2(C1)CN(C(=O)C(F)(F)CO)CCO2 23631,Cc1cccc(CCC(=O)NCC(CNC(=O)CCc2cnoc2)CO)c1Br 23632,N1(C(CCCNC(c2n(C=C)nnc2)=O)=O)CCC(N=[N+]=[N-])C1 23633,C(C)(CNC(=O)COCC1CCCC1)(CO)NC(C(C)OCCOC)=O 23634,N1(C(C=CCC)=O)CCN(C(C2CCCCN2N=O)=O)C(CCC)C1 23635,c1(C(=O)NC(C2CCN(C(c3cnco3)=O)C2)C)ccn2nccc2n1 23636,S(=O)(=O)(c1cc(C(N)=O)ccc1F)N(C)Cc1c[nH]nc1C(F)F 23637,C1(NC(c2cncnc2)=O)CCCC(NC(C2OCCCO2)=O)CC1 23638,CCCC(C)CN=c1[nH]c2c(c(=NC3CCC4(CC)CC34)[nH]1)CSC2 23639,N1(C(CC2CC(SC)C2)=O)CCN(C(=O)C(N)=O)C(C2CC2)C1 23640,C1(C#CC(=O)NC2CCC(C)N(C(c3cc(C)cs3)=O)C2)(CC)COC1 23641,c1(C(C)C)cccc(C(N2CCC(F)(C(=O)NC(c3ccccc3)C#N)C2)=O)c1 23642,O(C1CCOc2c(F)cc(F)cc21)C(=O)CCCCc1cnn[nH]1 23643,Cc1cc(C(N2CCCC2)C)c(O)nn1.c1(C(N(CC)C2CC2)=O)cnc[nH]1 23644,c1(CC)ncccc1C(=O)N(C)Cc1cncc(Br)c1 23645,N1(C(c2c(Cl)cn(CCC)n2)=O)CC(NC(=O)CSCC(C)C)CC1(C)C 23646,C=CCC(CC(F)F)NC(=O)CC1CCCCC1NC(C1CCCSC1C)=O 23647,c1(C(=O)N(C2CCCCC2)CCNC(C2(F)CCCC2)=O)cc(F)cc(F)c1 23648,C#Cc1cccc(C(N2CCN(CCNC(=O)CC3CCC(O)C3)CC2)=O)c1C 23649,C1(c2cn(CC(COC)O)nn2)(NC(=O)COC2(C)CCCC2)CC(F)(F)C1 23650,C(=O)(CCCCCC(C)(C)C)NC1CC2(C(NC(c3c(C)cc(N)cc3)=O)C2)C1 23651,C12(C(=O)NCC(C(C)C)OC)CCCC1CCN2C(C1CC2C=CC1O2)=O 23652,CC(C)C(C)CCNC(=O)C(C(C)O)NC(=O)CN1CCC(O)CC1 23653,Cc1ccc(Cl)c(O)c1C(N1CC(NC(C2CC(CF)C2)=O)CC(F)C1)=O 23654,N1(C(C(CC(=C)C)C)=O)CCC2(CC1)CN(C(c1ccc3scnc3c1)=O)C2 23655,C1(NC(C=C(C)C)=O)(CNC(=O)C(C)Cc2ccncc2)CCCCC1 23656,c1(C(N2C(C(C)(C)NC(C(F)=C(C)C)=O)CCC2)=O)cc2cc(Br)cn2cn1 23657,C(=O)(C(C)C(CC)CC)NC1(CC=C)CCN(c2nc(CC)nc(C)c2F)CC1 23658,Cc1cc(C(=O)N(C(C)CNC(=O)CC2CCCOCC2)C)cnc1O 23659,C1(NC(C(N2CCOCC2)C)=O)CC2(CCCN(C(C3C(C)C3C)=O)C2)C1 23660,C12(CNC(COCCCC)=O)CCC(CC1NC(c1ncccc1CSC)=O)C2 23661,N1(C(C(=O)N(C)C)=O)CC2CC(C1)C(CO)C2NC(C1CN2CCN1CC2)=O 23662,C1(C(N2CCCC(F)(c3ccccc3)C2)=O)COC2(CNC2)C1 23663,C12(CN(C)Cc3ccc(C#N)cc3)CC(C)(C1)OC21CCC1 23664,Cc1cccc(Cl)c1CN1CC(O)(CNC(=O)CC2CCOC(C(C)C)C2)C1 23665,N1(C(C(C)OCCN(C)C)=O)CCCCC(C(=O)NCCCc2nncn2C)C1 23666,CC(C)C1=NOC(C(N2CC(C)(NC(=O)COc3c(Cl)cccc3Cl)C2)=O)C1 23667,N1(C(C2C(C)C2)=O)CCCCC(NC(C2CC3CCC2CC3)=O)C1 23668,C#Cc1ccc(CC(=O)NC(C2CN(c3cc(C(F)F)ncn3)C2)C)cc1 23669,C1(NC(CNC(CC)=O)=O)CC2CN(C(c3cc(C)ccc3C)=O)CC12 23670,c1(OC)cccc(C(N2CCC(C(C)(C)NC(=O)CSC(F)(F)F)C2)=O)c1 23671,Cc1nn(CCF)cc1NC(=O)CCC1CCN(C(C2(C)CCCN2C)=O)CC1 23672,CN(C)NC(=O)CCC(=O)N1CCC(NC(C2CCS2(=O)=O)=O)C1C1CC1 23673,c1(C(N2CCC(O)(CNC(c3n(C)ccn3)=O)C2)=O)c(O)ccc2ccccc12 23674,C(=O)(C1CCCc2sc(=N)[nH]c21)N1CC(NC(C2CC(C)OC2)=O)CC2(C1)CC2 23675,c1(CNC(C(CC(C)C)O)=O)c(O)ccc(Br)c1O 23676,CC(C(=O)NC1(CNc2nc3ccc(F)cc3o2)COC1)C(C)S(C)(=O)=O 23677,c1(N2CCC(NCC(=O)N(CCOCC)C3CC3)C2)cccc(OC)c1 23678,c1(C(=O)NCC2(C)CCN(C(C34CCC(F)(CC3)C4)=O)C2)noc2ncccc12 23679,Cc1cc(CNC(c2coc(CNC(=O)CC3CCN(C)C3)n2)=O)sn1 23680,Cc1c(C(C)NC(=O)C(=O)N(C)C)oc2ccccc12.N12CCOCC(C1)C2=O 23681,CC1CN(C(=O)CC2(O)CCOCC2)CC1CC(N1CCC1CF)=O 23682,CC(C(F)(F)C(F)(F)F)=CC(N1CCC(NC(c2cc(C)nc(O)c2)=O)C1)=O 23683,N1(C(C(C2CCCC2)OC)=O)CCCC(O)(CNC(=O)C=Cc2cscn2)CC1 23684,c1(C(c2nnnn2C2CC2)NC(C2CCCC2)C2(CCOC)CC2)cc(Cl)no1 23685,Cc1oc(CO)cc1C(N1CCN(C(C2CNC(=O)C2)=O)CC1)=O 23686,N1(C(Cc2cnc(C)[nH]2)=O)CC2CCC1C1CN(C(=O)C=CC3CC3)CC21 23687,C1(CCNC(CN(C)C2CC2)=O)CCN(C(C2CC3C(C2)C3(F)F)=O)CC1(F)F 23688,C(C#N)(C(C)CC)c1scc(C(N(CCCC)Cc2cnoc2CC)=O)n1 23689,C1(C(N2CCC(n3cc(C(C)N(C)C)nn3)CC2)=O)CCC2(CCC2)C1 23690,C12(CNC(CCN(CC)CC)=O)CCN(C(=O)CC(C)(C)C)CC1C2 23691,c1(OC)ncnc(C)c1C(=O)NCC1CCN1C(C1CC(F)(F)C1)=O 23692,c1(C(=O)NC(CNC(C(C)(CO)NC(C)=O)=O)C2CCC2)ccc(C)c(C)c1O 23693,c1(C(=O)NCC=CCC(=O)Nc2cnn(CC3CC3)c2)cc(C(F)F)no1.C 23694,C1(C(=O)NCC2=CCN(C(C=CC(C3CCCC3)=O)=O)CC2)CCC2(CCOC2)O1 23695,c1(C(=O)NC(C(=O)N(CC(C)O)CC2CC2)C)cc(CO)on1 23696,C1(O)(CNC(c2c(COC)ncs2)=O)CCN(C(C2CNC(=O)N2)=O)C1 23697,Cc1occc1C(=O)NCCC(C)NC(c1cnsc1C)=O 23698,c1(C(C)C)nnc(C(=O)NC2CC(n3ccnn3)C2)o1 23699,N1(C(c2ccc(OC)c(F)c2F)=O)CCCC2(CCCN2C(C2C=CCC2)=O)C1 23700,N1(C(c2cc(C)nc(C)c2)=O)CC(C)CN(C(c2nc(Cl)sc2Cl)=O)C(C)C1 23701,N1(C(c2cnc(OC)s2)=O)CC2CCC1C(CNC(=O)CCCC(N)=O)C2 23702,Cc1cc(Br)ccc1CCC(=O)NC1CCCC(NC(=O)C2=COCC2)C1 23703,c1(C(=O)NCCN(C(=O)CC(O)c2ccccc2)CCOC)nocc1C 23704,C1(CC(=O)NCCC2CCN(C(C3(C)CCCC3)=O)C2)CCCC1(F)F 23705,C1(Cc2c(CNC(C3CC(CCC(=O)NC4CC4)C3)=O)ocn2)CC2CC1CC2O 23706,N1(C(C2(C3N(C(C4CCCCCC4)=O)CCC3)CC2)=O)CCN2CCCCC1C2 23707,c1(C(N(c2cc(C)c(Cl)cc2)C)=O)ccc2c(c1)COC2 23708,N1(C(c2ccc(C)o2)=O)CCCC(C)(C(N2CCCC2c2ccc(Br)cc2)=O)C1 23709,c1(N2CC3CC(NC(c4cccc(C(C)C)n4)=O)C3C2)ncnc2c1CCO2 23710,N1(C(CCC=C)=O)CCC(NC(c2cc(C(C)C)n(C)n2)=O)C(CC)C1 23711,N1(C(C(CC)n2cccn2)=O)CCC(O)(Cn2cc(CO)nn2)C1.C12(CC1)C(=O)N2 23712,N1(C(=O)Nc2n(C)nc(C)c2Br)CCCc2ncccc2C1 23713,C(C(=O)NOCCN(C)C)N(C(=O)CC1(C)OCCO1)C(C)C 23714,c1(OC)cc(F)c(S(=O)(=O)NC2CCCC2P(C)(C)=O)cc1OC 23715,c1(CC(=O)NC2CC(NC(C(n3cc(C)nc3)(C)C)=O)C2)cccc2nonc12 23716,S(=O)(=O)(c1c[nH]c(C(=O)NC2CCN(C(=O)C(C)(C)C#N)C2)c1)NCC 23717,N1(C(C(C)c2ccsc2)=O)CCCC(O)(CCNC(=O)C(C)(Cl)Cl)C1 23718,C(=O)(C(O)CC(F)F)N1C(CNC(Cn2nc(C)c(Cl)c2)=O)CCC1 23719,C(=O)(C1=CCC(NC(c2cnn(C)c2Cl)=O)C1)NC(C1CC(F)(F)C1)C 23720,CC(C)(C)C(CN=c1ccn2c(Br)cnc2[nH]1)NC(c1ccc(F)o1)=O 23721,N1(C(Cc2scc(C)c2)=O)CC2(CNC(=O)C(C)n3cncn3)CC1CO2 23722,C12(CNC(CC3C(C)(C)C3)=O)CC1CN(C(=O)CCCc1ncc(Br)cn1)C2 23723,C1(C(=O)NC2CCC(CCCC)C2)CCNC(C2CC2)C1 23724,N1(C(Cc2ccc(C)nc2)=O)CC(C)(C)C(NC(c2cccnc2)=O)C(C)(C)C1 23725,C(CSC)(C(=O)NCCCOCCCNC(=O)C=CCc1ccccc1)OC 23726,N1(C(=O)OC(C)(C)C)CC2COCC2(C(=O)NC(C)(C)CN2CCOCC2)C1 23727,c1(C(=O)NC2C(CNC(C34CCC(OC)C3C4)=O)C2)[nH]c2ccccc2c1C 23728,C(CN=c1nc2sccc2c(NCCCC(F)(F)F)[nH]1)N1CC(CC)OCC1 23729,c1(CC(=O)NCC2CCN(C(C3ON=C(C)C3)=O)C2)ccc(F)cc1[N+](=O)[O-] 23730,C1(OCC)CCCN(C(c2nc(CNC(C3CC(C)=NO3)=O)cs2)=O)C1 23731,C(=O)(C(C)(C)CC(C)=O)NCC1OCC(C(=O)NCC(C(CC)C)(C)O)C1 23732,C1(CC(=O)NCC2(F)CN(C(C3(C)CCCOC3)=O)C2)CN2CCN1CC2 23733,CC1(C)CN(C(=O)CCc2nccs2)CC1CNC(c1cc(CO)[nH]n1)=O 23734,N1(C(C(C)OCCCC)=O)CC(C(N2CC(C(C)(C)O)C2)=O)CC(C)C1 23735,C(=O)(C#CC1CCCCO1)NCCN(C(C)C)C(c1ccc(OCCF)cc1)=O 23736,c1(C(N2C(C(C)NC(C3CC(C#N)C3)=O)CCCC2)=O)cc2cc(F)ccc2o1 23737,CCCCC(F)C(=O)N1CCCCC1C1CCN(C(=O)Cc2ccc(F)cc2)C1 23738,NS(=O)(=O)c1ccnc(C(=O)NCC2CN(C(C3CNC(=O)N3)=O)CC2(F)F)c1 23739,Cc1ccc(C(F)(F)F)cc1NC(=O)COC(F)F.C1C(CC(C)C)C(=O)N1 23740,C1(C(N2CCC(CC=C)(NC(c3cnc(Cl)[nH]3)=O)C2)=O)CCC(N=[N+]=[N-])CC1 23741,N1(C(COCCCC(C)C)=O)CCC2(C1)CN(C(C1CC1C(F)F)=O)C2 23742,CCC(O)CCN=c1[nH]c(N2CCN(CCCOC)CC2)nc2cccnc12 23743,c1(CC)nc(C(N2CCC(C(C)NC(c3cncs3)=O)C2)=O)co1 23744,c1(C(=O)NC(CC(C)NC(=O)Cn2ccnn2)C)ccc(-c2csnn2)cc1 23745,N1(C(c2ccc(C)nc2)=O)CCC2C(C1)CN2C(=O)CCn1ccc(O)nc1=O 23746,C(CC(C)C(=O)N(C)CCNC(c1c(C)nsc1I)=O)OC 23747,C12(NC(C=CC(=O)OCC)=O)CC1CN(Cc1cccc(CO)n1)C2 23748,C1(CC(=O)NCc2cccc(O)c2)CCCCN1C(=O)CN1C(=O)CNC1=O 23749,C1(NC(C2C(=O)NCCCC2)=O)CC2CC(C1)N(C(c1ncoc1C1CC1)=O)C2 23750,C12(NC(C3CN(C(CCC=C=C)=O)C(CO)C3)=O)CC3CC1C2C3(F)F.C1C(=O)N1 23751,N1(C(C(COC)C)=O)CCC2(CCC(NC(C3CCC(F)C3)=O)CC2)CC1 23752,c1(C(=O)NC(C)CNC(=O)CC2CC3CC3C2)c(Cl)csc1Cl 23753,CC1CN(C(C2(c3ccccc3F)CC=CC2)=O)CC1NC(=O)CCF 23754,C(=O)(C(CCC)N(C)C)NCC(C)(C)NC(COCCOCC=C)=O 23755,C(=O)(CC(C)C(C)(C)NC(C1CC(C)(CC)C1)=O)NCC1(CO)C(C=C)C1 23756,N1(Cc2c(CC)noc2)CCC(CNC(c2nccnc2CN(C)CC)=O)CC1 23757,c1(CC(=O)N(C(C)C(C)(C)O)C)ccc(NC(=O)OC(C)(C)C)nc1 23758,C1(NC(C(C)(C2CC2)NC(C)=O)=O)CN(C(=O)Cc2ccc(CO)cc2)CC1O 23759,c1(C(=O)NC(C(C)NC(C2C=C(C)CS2)=O)C)cn2cccnc2n1 23760,c1(C(=O)NCC2=CCN(C(C(=O)NC)C)CC2)noc2ccccc12 23761,c1(C(N2CC3(CCN(C(=O)CCC4CC4)C3)C2)=O)ccc(Cl)c2cccnc12 23762,c1(OC)ccccc1OCC(=O)NC(CNC(c1cn(C)nc1C)=O)C1CCC1 23763,CC(CC(=O)N1CCC(CNC(=O)C(c2cc(F)cc(F)c2)O)C1)C(F)(F)F 23764,c1(C(N2CCN(C(=O)C#CC3CCCOC3)CC2)=O)cnc2ncnc(O)c2c1 23765,Cc1ccc(C2(C(=O)NCc3c[nH]c(C#N)c3)CC2)cc1.C12CCCN1C(=O)N2 23766,C(C(C)(C)C(F)(F)F)C(N1CC(C(C(N2CC(CC(=O)OC)C2)=O)OC)C1)=O 23767,CC1=C(C(=O)NC2CC3CC(NC(=O)C(O)CN(C)C)CC23)SCCO1 23768,N1(C(c2nn(CC)c(O)c2)=O)CCC2(CC1)CC2CNC(=O)CC(O)CC(C)C 23769,C1(C(=O)NCC2C3CN(C(C4(C)CCCCC4)=O)C2C3)CS(=O)(=O)CC(=O)N1 23770,O=C1CCN(C(C23CC(CO2)N(C(=O)C(C)(C)C2CCCO2)C3)=O)CCN1 23771,N1(C(c2c(C)nc(O)[nH]2)=O)CCC(NC(c2cc(C(F)(F)F)no2)=O)CC1C 23772,CC1CC(C(N2CCCC(N(C(=O)Cc3cncc(O)c3)C)CC2)=O)CC(C)C1 23773,N1(C(C2(OC)CC(C)C2)=O)C2CCC(C(=O)NCc3cnns3)C1CC2 23774,C(CCCCC(=O)NC1CCC(C)N(C(c2[nH]nnc2C2CC2)=O)C1)NC(C)=O 23775,Cc1nn(CC(=O)NCCCC(=O)NCCC2CCCO2)c(=O)o1 23776,C1(CNC(C2C(=O)NCC2)=O)CC2CC2N1C(c1ccn(CC(F)F)n1)=O 23777,n1(CC(=O)NCC(CNC(C2CC3CCC(C2)O3)=O)OC)nc(C)c(C)c1C 23778,C1(NC(C2(C)CC(NC(c3c(C)noc3)=O)C2)=O)CCOC2(CCC2)C1 23779,C1(O)(CN(C(=O)C(F)=C2CCC2)C)CCN(C(c2ccc(C(C)(C)C)[nH]2)=O)C1 23780,c1(C(=O)NCC2CCC(NC(C3C(C)CCC3)=O)C2)cc2c(F)c(F)ccc2[nH]1 23781,c1(N(C)C)ccc(C(=O)NC(CNC2CCC(=O)N2)C2CC2)cc1[N+](=O)[O-] 23782,c1(C(N(C2CCN(C(c3conc3C(C)C)=O)C2)CC)=O)cc(C(F)(F)F)co1 23783,C1(F)(CNC(c2ccc(C#C)cc2OC)=O)CC2CCC(C1)N2C(=O)C=C(C)C 23784,Cc1cc(C)n(-c2ccc(-c3nc(-c4ccn(C)c4)n(CCC(C)C)n3)nc2)n1 23785,c1(C(N(CC(C)O)CCNC(CCC#C)=O)=O)cnc2c(c1)CNC(=O)N2 23786,C(=O)(C(O)CCNC(=O)C(O)C1CCCC1)NC(C1CCCC1O)C 23787,C1(CN(C(C=CCN(C)CC)=O)C)COCCN1C(=O)C=C1CC1 23788,N1(C(C(CSC)C)=O)CC(NC(=O)C(CO)NC(=O)C(F)(F)F)CC(F)C1 23789,c1(SC(C(=O)NC2CC(CNC(Cn3nnc(C)n3)=O)C2)C)ccc(C#N)cc1 23790,N1(C(C=CC=CCC)=O)CC(NC(c2cnc(C)nc2CC)=O)CCC1C 23791,CC(C)CC(F)C(=O)NCC1(C)CN(C(=O)CCCN2CCCCC2)CC1C 23792,N1(C(C(C)C(C)(F)F)=O)CCCC2(CCCN2C(c2cnc3ccccn23)=O)C1 23793,C1(COC)(NC(C23CC4CC2C3C4)=O)CCN(C(=O)C(c2ccc(O)cc2)F)C1 23794,N1(C(c2c(C)nc(C)s2)=O)CC2(CC(NC(c3n[nH]c(C)c3[N+](=O)[O-])=O)CO2)C1 23795,c1(OC)cc(Br)c(C(=O)COC(c2cc3c(s2)CCNC3)=O)cc1OC 23796,N1(C(c2c(CC)nc(C)[nH]2)=O)CC(NC(C2(C)CCN(C)C2)=O)CC12CCC2 23797,c1(CC)cc(C(=O)NC2(C)CC(NC(=O)C(C3CC(F)(F)C3)OC)C2)ccc1C 23798,c1(CC(=O)NCC(CNC(CC(=O)OC)=O)OC)ccc2ncsc2c1 23799,C1(CN2CCC(C=C)C2)CN(C)CCN1C(c1cc(OC)cc(F)c1)=O 23800,N1(C(CC(C=C)CC)=O)CC(C)CN(C(=O)CCCc2cnn[nH]2)C(C)C1 23801,N1(C(Cc2ccc(C)s2)=O)CCC(C2CC2)C1CNC(=O)COc1ccsn1 23802,c1(C(=O)NC(C)CC(C)NC(=O)C(C)(C)c2ncco2)ccc([N+](=O)[O-])c(N)n1 23803,CCC(CC)CC(F)C(=O)NCCC(C)(C)C(=O)NCC1(C)CCN(C)C1 23804,CC(C(=O)NC1C=CC(C(=O)NC(C)C(=O)NCCF)C1)C(F)F 23805,C1(OC)CC(CNC(c2csnc2C)=O)N(C(C2CC(N(C)C)C2)=O)C1 23806,C(=O)(C(C)S(N)(=O)=O)N1CC(c2cn(C(COC)COC)nn2)(O)C1 23807,N1(C(C2(C#N)CCC2)=O)CCC2(CCCC2NC(C23CCCC2C3)=O)CC1 23808,CCCC(C(O)C(=O)NCC1(O)CCCOC1)NC(c1ccccc1CC)=O 23809,N1(C(c2ccc(OC)cc2F)=O)C2CCC1CC(NC(=O)C(C)CS(C)(=O)=O)C2 23810,C=CCCCC(C(=O)Nc1cccc2c1CCO2)NC(=O)CC1C=CCCC1 23811,c1(C(=O)OC)cnc(C(C)C)[nH]c1=NCCCC(C)(C)NC(=O)CC(C)SC 23812,N1(C(c2c(N)cnc(Cl)c2)=O)CCCC(NC(=O)Cn2cc(CO)nn2)C(F)C1 23813,C(C(C)(C(=O)NC(CNC(c1cc(Cl)c[nH]1)=O)C(C)C)OC)OC 23814,c1(CC(N2C(CCN(C(CC(CC)SC)=O)C)CCCC2)=O)ccc(C)c(C)c1 23815,Cc1c(C(N2CCC3(CC3C(=O)Nc3cc(O)ccn3)C2)=O)ccc(Br)c1F 23816,C1(CC=C)(C(=O)NC2CC(C(C)NC(c3cscc3Cl)=O)C2)CCOC1 23817,N1(C(C2(C)CCOC2)=O)CCC(C(F)F)(CNC(c2ncc(F)cn2)=O)C1 23818,C1(=O)C(C)CN1C.C(C)(CCOCCSCO)N(C(C)=O)C.C(C)(C)(C)O 23819,C1(C(=O)NCC2(O)CCN(C(c3c(C)cc(F)s3)=O)C2)SC2C=CC1CC2 23820,C#CC1(O)CCN(C(c2cnc(CNC(=O)C(C)(C)C(O)CC)nc2)=O)CC1 23821,c1(C(=O)NC(C(C)NC(C(C)NS(CC)(=O)=O)=O)CO)cccc(N)c1F 23822,c1(C(=O)NC(C)C(C)(C)NC(=O)CC2COCCN2C)cccc(C(C)(F)F)n1 23823,N1(CC(=O)NCC2(CC(=O)N(CCOC)CC3CC3)CC2)C(=O)CCCC1=O 23824,Cc1cncc(C=CC(=O)NC2CC2NC(=O)C(c2cc(Cl)ccc2Cl)(F)F)c1 23825,Cn1cnc2nc(N3CCC(NC(=O)C=CI)C34CCCC4)ncc12 23826,Cc1nc2cccc(C(N3CC(CNC(C4(CCO)CC4)=O)C4(CC4)C3)=O)c2s1 23827,C(=O)(C(C(F)(F)F)=Cc1ccccc1)NC(C)CNC(c1cc(C(N)=O)no1)=O 23828,N1(C(C(CCC)=CCC)=O)CCCC(N(C)C(C2(c3ccno3)CCC2)=O)CC1 23829,Cc1cc(NCCCC(C)NC(C2CC2F)=O)ccc1NC(=O)C1=CCCC1 23830,C(=O)(C(C)(CC1CCC1)OC)NCC1C(NC(CCNS(CC)(=O)=O)=O)CC1 23831,Cc1nnc2ccc(C(N3CCC(NC(=O)CC4(C)CC4(Cl)Cl)C3(C)C)=O)cn12 23832,c1(C(N2CCC(C(C)NC(C=C=C(C)C)=O)C2)=O)cccc2c[nH]nc12 23833,C(=O)(CC(O)CC(C)C)NCCN(CC(C(C)C)OC)C(=O)COCC(C)(C)C 23834,C1(CC(=O)N(CCOCC)C)CN(C(=O)CC2(COC)CCOCC2)CCO1 23835,Cc1nn(CC(=O)NC2CC3C(NC(=O)C(c4cnccn4)C)C3C2)c(=O)o1 23836,c1(C(C(N2C(CN(C(C(F)=CCC)=O)C)CCC2)=O)O)ccccc1F 23837,N1(C(C(C(C)O)(C)C)=O)CC2COCC2(C(=O)NCc2ccc(Cl)cc2)C1 23838,c1(C(C(=O)NCCCN(C(=O)C(O)c2ccsc2)CC)C)c(F)cccc1F 23839,C1(C)(C(N2CCN(CCCNC(C(C(C)C)F)=O)CC2)=O)CCCCC1(F)F 23840,C1(C(=O)NCCOC2CCN(C(C(C)NC(C)=O)=O)CC2)CC(C(C)C)=NO1 23841,C(C(CCC)C(=O)N1CCC1(C)CC)NC(C(C=C)O)=O 23842,c1(C(N2CCN(C(CC(C=C)C)=O)CC2C2CC2)=O)ccn2ncc(C)c2n1 23843,N1(C(C2C(CCC)C2)=O)CC2(C)CC1C2NC(c1ccc(=O)n(CC(C)O)c1)=O 23844,C(C)(C)(C(=O)N1CCC(C(C)NC(c2cccnc2)=O)C1)SC 23845,c1(C(=O)NCC2CC(C)N(C(=O)CC3C=CCC3)C2)ncc(Cl)cc1Cl 23846,c1(C(=O)NC2C(CCC(C)C)CCC2)ccc(F)c2cccnc12 23847,c1(CC)ncsc1C(=O)NC1(CN(C(=O)CC(F)F)C)CC1 23848,CCCCC(Cc1ccccn1)NC(=O)NC(c1cccnc1)c1cccnc1 23849,C1(C(N2CC(N(CCCOC3CC3)C)C2)=O)CC(C)(C(C)(C)C)C1 23850,N1(C(C(CC=C)(F)F)=O)CCC2CN(C(=O)CC3CCCN3C(C)C)CC2CC1 23851,C1(NC(CCOCC)=O)CC2CCC1CN2C(C1(C#N)CCOCC1)=O 23852,Cc1c(NS(=O)(=O)c2cc(Br)c(Br)cc2F)cc([N+](=O)[O-])cc1[N+](=O)[O-] 23853,CCC(C)C(O)C(=O)NCC1(NC(=O)C2=NOC(C3(O)COC3)C2)CCCC1 23854,c1(C(=O)NC(C(CO)NC(c2cccc(C(C)=O)c2)=O)C)onc2c1CCCC2 23855,N1(CC2CCC(C(=O)OCC(C)C)CC2)CCC(CO)C(F)(F)C1 23856,C=CC(C)CC(=O)NCc1ncn(C(C)C)n1.C12(OC)CN(C1)C(=O)C2 23857,c1(C(=O)NC(CNC(COCCOC)=O)C)ccc(SC(C)(C)C)cc1 23858,c1(OCC)nc(Cl)cc(=NC(=O)C2CC(F)CN2Cc2cccc(I)c2F)[nH]1 23859,c1(C(N(CC)CC2CCCN2C(=O)C=CS(C)=O)=O)cnn2cccnc12 23860,c1(C(N2CC(C)(CNC(c3c(C)c[nH]n3)=O)OCC2)=O)cc2c(s1)CCCC2 23861,c1(C(N2CCN(Cc3c(C)n[nH]c3C)CC2)=O)ccc(O)c(C(=O)C(C)C)c1 23862,S(=O)(=O)(c1cccnc1[N+](=O)[O-])N(C)CP(C)(C)=O 23863,c1(C(=O)NC2C(NC(=O)Cn3nccn3)C2)ccc(SC(F)(F)F)s1 23864,N1(C(CCOCC)=O)CC(CNC(=O)CN2CCSCC2)CC(C)(C)C1 23865,C1(O)(C(C)NC(Cc2c(C)scc2)=O)CCN(C(c2n[nH]c(C3CC3)c2C)=O)C1 23866,C1(C(=O)NCC(CNC(C2(CCOC)CC2)=O)C)Cc2cc(F)ccc2O1 23867,C1(C)(CNC(CCNC(Cc2c(C)noc2C)=O)=O)CC2CCC1C2 23868,N1(C(=O)C=O)CC2CCC1C(C)C2.N1(N2CCC(C(F)(F)F)C2)CCS(=O)CC1 23869,C1(N(C)C(c2ccc(C3CC3)o2)=O)CCC2CN(C(=O)Cc3nccn3C)CC12 23870,S(=O)(=O)(c1cnccc1N1CCS(=O)(=O)C(CO)C1)NC(c1ccc(Br)cc1)C 23871,C1(NC(CC=C)=O)CN(C(=O)CCC2CC2C)Cc2nccn2C1 23872,c1(C(N2C(CNC(C3(C)CC=CCC3)=O)CC2)=O)c(N)cc(F)c(Br)c1F 23873,c1(NC(CC)CO)cc(Br)ccc1S(=O)(=O)NC1CCCN(C)C1 23874,CCCC(CCCO)C(=O)N1CCCC(C2CC2NC(=O)COC(C)C)C1 23875,C1(C2CCOCC2)(Nc2cccc(Cn3c(C)csc3=O)c2)CC1 23876,CCC(c1cccc(Cl)c1)=CC(=O)NCCCCN(C)C(C1CCCN1CC)=O 23877,C(=O)(C(O)CCCC)NC(C1(O)CCN(C(CSCCC)=O)C1)C 23878,N1(C(C(C2CCCC2)OCC)=O)CCC(CNC(c2cnc(O)o2)=O)CC1C 23879,N1(C(CCNS(CC)(=O)=O)=O)CCN(C(=O)Cn2c(C)c(C)sc2=O)C(CO)C1 23880,Cc1cc(C(=O)NCC(C)(CC(C)C)NC(=O)C(C)Cn2ccnc2)c(C)cn1 23881,Cc1cc(C(=O)NC2CCCC(NC(c3ncc(C)cc3Br)=O)C2)cc(F)c1 23882,N1(C(c2nc(C)n(C)c2C)=O)CC(C)OC2(CCN(C(=O)CCCC(C)C)C2)C1 23883,N1(C(CN(C)C(C23CC(CO)(C2)C3)=O)=O)CC=CC12CCOCC2 23884,C(=O)(CS(=O)C(F)(F)F)N1CCC(NC(C(CC)=CCCC)=O)CC1C 23885,c1(C(=O)NCC(CC)NC(c2cn(CCF)nn2)=O)c(OC(F)F)cccc1F 23886,c1(C(=O)NCC2(NC(CCC=C)=O)CCC2)sc2nc(C)nc(C)c2c1C 23887,Cc1ccc(-n2ccnc2)c(C(=O)NC2C=CCN(C(C3CC3C)=O)C2)c1 23888,c1(OCC(N2CC(C3CCN(C(=O)C(F)=CCCF)CC3)C2)=O)cccc(O)c1 23889,Cc1cc(C(=O)NC2CC(CNC(C3CCCN3C3CC3)=O)C2)cc(C)c1C 23890,CC1=CC2CCCC(C1)N2C(=O)NCCCNC1CCC1 23891,CC#CCC(C(=O)Nc1ccc(O)cc1C)NC(=O)C(C)NC(N)=O 23892,C1(NC(CCC(C)OC)=O)CC2CCC(C1)N2C(=O)C(=Cc1cnn(C)c1)C 23893,c1(C(N(CCN(C(C(CCCOC)C)=O)C)C)=O)cccc2c1C1CCC2CC1 23894,N1(C(C2(C(C)NC(C(C(CC)C)OC)=O)CC2)=O)CC2C=CCC(C2)C1 23895,c1(OC)c(Cl)nc[nH]c1=NCC1CCCN(C(c2cnn(C)c2N)=O)C1 23896,C12(C(=O)NCc3ccc(C)c(Cl)c3)CCC(CC1)N(C(=O)C(O)CC(F)(F)F)C2 23897,c1(NCC(C2CCCCC2)NC(C2C(C)(Br)C2)=O)cnc2ccccc2n1 23898,S(=O)(=O)(c1ccc(N2CCC(O)C2)cc1Br)N(C)C1CC1.CCC1CNC(=O)N1 23899,c1(NC(C(C)(C)CCl)c2n(C)nnn2)ccc(Cl)c(C(N)=O)c1 23900,N12CC(C(C)C1)NC2=O.CCCCCCSc1cc(-c2ccncc2)n[nH]1 23901,CCS(=O)(=O)CC(=O)N1CCC(NC(=O)CCCOC(=O)CCC)C1.C(C)(C)C 23902,c1(OC)ccccc1C(C)(C)C(=O)NCC(C1CC1)NC(C1CCCS1(=O)=O)=O 23903,c1(N(C)CC2(NC(=O)CNS(=O)(=O)C3CC3)CC2)ncc2c(ncn2C)n1 23904,N1(C(C(CCCC)C)=O)CCCC2CN(C(C3CN(CC(C)C)C3)=O)CC12 23905,C1(C(=O)NC(c2ccn(C)n2)C)(NC(Cc2c(C)ccs2)=O)CCN(C)C1 23906,C(C)(C(=O)N1CCCC(C)(CNC(=O)CCC2CCCCC2)C1)(C(C)C)OC 23907,N1(S(c2c(N3CC(CC)SCC3)nccc2)(=O)=O)CCc2cc(C)cc(C)c2C1 23908,C1(CNC(c2n(CC)ncc2)=O)CC(OC)CN1C(c1cn(C2CC2)nn1)=O 23909,C(=O)(C1=CCCOC1)NC12C(CN(C(C(C)(C)CC3CC3)=O)C1)C2 23910,c1(C(=O)NCC2N(C(C(C(CC)C)O)=O)CC(F)C2)c2n(c(=O)n1C)CCCC2 23911,Cc1ccc(C(F)C(=O)NCC(=O)NCC2CCOCC2)cc1 23912,Cc1nccc(CCC(=O)NCC2CCCCN(C(C3(C)CCCCO3)=O)C2)n1 23913,CCCCC(C(=O)NC)NC(C12CC1CN(C(c1cc(C)ccc1O)=O)C2)=O 23914,c1(N(CCC)C(=O)NC2CC2c2cnco2)ncc(OC)cc1C 23915,n1(C(CC)C)ccc(=NC(=O)c2ccc(C3CCCN3)s2)[nH]1 23916,C1(C(=O)NCC2N(C(C)=O)CCC2)CN(C(C2CCOC2C)=O)CCO1 23917,C(=O)(CCCCC(F)F)N(CCNC(c1nc(COC)sc1)=O)C(C)C 23918,C(=O)(C#CC(C)(C)C)N1C(C)(C(=O)NCCCCC)C=CC1 23919,CC(CN=C(NCC1(N2CCCC2)CCCC1)NC1CCCC1)CC(F)(F)F 23920,N1(C(C2CC(SC)C2)=O)CCC(NC(C2CCN(CC(C)C)C2)=O)C1C 23921,C(=O)(CCC(F)(F)F)NC(C1(O)CCN(C(c2nn(C)cc2Cl)=O)C1)C 23922,C1(C)(NC(CCOc2ccc(C)cc2)=O)CCN(C(C2CC=CCC2)=O)CC1 23923,c1(OC)cc(CCNC(=O)C(F)(F)c2ccncc2)ccc1I 23924,N1(C(C(C)(N(C(COCC(C)C)=O)C)C2CC2)=O)CC2CCC2(CO)C1 23925,N1(C(C(C2CCOC2)OC)=O)CC(C)(NC(=O)COC2CCCCC2)C1 23926,C(=O)(C(F)C(C)CNC(c1cncc(OC)n1)=O)NCc1n(CC)cnn1 23927,c1(OCC(=O)NCCCNC(C(C2CCOC2)OCC)=O)ccccc1C 23928,N1(C(CCC(=O)OC(C)(C)C)=O)CC2(C1)CN(C(c1cnn(CCF)c1)=O)C2 23929,N1(C(c2c(C)nn(C)c2C)=O)CC(NC(=O)Cc2nncs2)CC2(CC2)C1 23930,C1(CNC(c2c(COC)cco2)=O)C2CCCC1N(C(=O)Cc1csnc1C)C2 23931,CCCCCCCC(F)C(=O)N1CC(O)(CNC(C2CC3CCC2O3)=O)C1 23932,Cc1c(C(N2CCCC2C(C)NC(C2CCCN2C)=O)=O)cnn1CCO 23933,S(=O)(=O)(c1cccc(S(N)(=O)=O)c1)NC(c1ccc(C)c(S(N)(=O)=O)c1)=O 23934,N1(C(C(C)N(C(=O)C2=NOCC2)C)=O)CC(F)CC1C 23935,C1(OCCC)CN(C(=O)Cc2[nH]cnc2C)CC1NC(C(N1CCC(C)C1)=O)=O 23936,C(CNC(=O)Cc1c(Cl)cnn1C)(CCCC)NC(CSCC=C)=O 23937,C(c1ccc(F)cc1F)=CC(=O)NCCC1(NC(C(CCSC)OC)=O)CCC1 23938,C(=O)(CCCCC(=O)OC(C)(C)C)N1CC=CC(NC(C2CC(C)OCC2)=O)C1 23939,C(=O)(C1=CC2CCC(C1)C2)N(CC(CC)NC(C1CCC([N+](=O)[O-])CC1)=O)C 23940,C(C)(C)(CCN=c1nc(C#N)[nH]cc1Cl)NC(c1ccc(OC)cn1)=O 23941,C1(C(=O)Nc2nc(-c3ccccc3)cs2)CN(C(c2sccc2F)=O)CCN1 23942,C1(C(=O)NC2CC(NC(Cn3c(C)ccc3C)=O)C2)CC(S(C)(=O)=O)C1 23943,Fc1ccccc1C(F)(F)C(C1CCC1)OCCC1CCO1 23944,c1(C(N(CC(CNC(COC(C)=O)=O)C)C)=O)c(Br)c(C)nn1C 23945,CC1SCCCC1C(=O)NC1CCN(C(=O)C=Cc2cnccn2)CC1 23946,N1(C(C(C)(C)O)=O)CCC(C2CCN(C(C3(C(F)F)CC(O)C3)=O)CC2)C1 23947,N1(C(CCCOCC=C)=O)C2CCC1C(C(N1CCC(C(C)CO)CC1)=O)C2 23948,N1(C(CCSCCC)=O)CCN(C(=O)Cc2nocc2C(C)C)CCC1C 23949,C=CC(CC)CC(=O)NCC1(O)CCN(C(c2cnc(C)c(OC)c2)=O)C1 23950,CCC(C)CCC(=O)N1CCC(CNC(c2cncnc2C)=O)C1(C)C 23951,C(C)(C(=O)N(CC(=O)NC(C)CN1CCCC1)CC1CC1)OCC(C)C 23952,C#Cc1cc(NC(C2CC2CC(C)C)=O)ccc1C.C1C(N(C)C)C(=O)N1 23953,Cc1ncccc1CCNC(=O)CCOCCNC(=O)Cc1ccc(O)cc1 23954,C1(C(C(=O)NCCC(=O)OCC)N(CC(C)SC)C)CCCC(C(=O)OC)CC1 23955,C1(NC(C(CC#C)C)=O)CN(C(c2ccc3scnc3c2)=O)CC12CCOCC2 23956,c1(C(=O)NC2CCN(C(C3(OC)CCC3)=O)CC2)cnc2nc(C)ccc2c1O 23957,N1(C(C2C(C(=O)OC)CCCC2)=O)CCOC2(C1)CN(C(C1(O)CCCC1)=O)C2 23958,c1(CNC(C2CC(c3ccc(O)cc3)C2)=O)cc(Br)cc2c1OCC2 23959,C1(NC(c2ccn(C(C)C)n2)=O)CC(C(N2CC(O)(C(N)=O)C2)=O)C12CCC2 23960,c1(C(N2CC(NC(C(C)=CC)=O)C3(C2)CC3)=O)cc(Br)cc(C)c1OC 23961,Cc1ncnc(C(N2CCCC(NC(C3(F)CCCOC3)=O)C2)=O)c1C 23962,Cc1noc(C)c1CC(C)C(=O)N(C)CC1CN(C(C2CC3C=CC2C3)=O)C1 23963,N1(C(c2cc(C)c(C)o2)=O)CCC(C)(CNC(=O)CCNC(C2CC2C)=O)CC1 23964,C1(CCC)COCCN1C(=O)CNC(=O)CNC(C1C2CCCOC12)=O 23965,C(N=c1[nH]c2ccc(Cl)cc2c(=NCC(F)CO)[nH]1)c1ccc(OC)c(C)c1 23966,CCC(C)(C)CC(=O)NCc1ocnc1C(=O)Nc1cc(OC)ccc1O 23967,n1(CC)cc(C(=O)NC(c2cccnc2)C(=O)NCC2CCCS2)c(C)n1 23968,C(=O)(CCCCC#N)N1CCC(F)(CNC(C(C)Oc2ccccc2F)=O)C1 23969,c1(NC(CNC(C2CC(=C)C2)=O)=O)ccc(CCCC)nc1 23970,C(=O)(NNC(=O)N1CCCC1C(F)(F)F)c1n(C)ncc1 23971,c1(CCC)cccc(C(=O)NC(C)CCCNC(=O)CC2CC3(CC3)C2)c1 23972,N1(C(C2(OC)CCC2)=O)CC(CC(=O)NCCn2nc(C)cc2C)C2(CC2)C1 23973,c1(C(=O)NCC2C(C)CCN2C(C2CN(C)C2)=O)cccc2nncn12 23974,CC(C)C(C)(C)C(=O)NCc1cc(C(=O)NC(C2(CO)CC2)C)n[nH]1 23975,O=S(=O)(c1ccc(NCc2cc(F)ccc2F)cc1Br)NCCC1(CO)CCCC1 23976,C1(C2C(C#N)CC2)CCC2(CC1)CC(NC(=NCCN=[N+]=[N-])NC1CCOCC1)C2 23977,c1(SCC(=O)NCC2(OC)CCN(C(C(CC)SC)=O)C2)nc2ccccc2[nH]1 23978,c1(CN2CCN(C(c3c(C)ocn3)=O)C(C)C2)sc2ccccc2c1Cl 23979,CC1(C)CCCC(CC(=O)NCC(C)(F)CNC(C2CC(O)C2)=O)C1 23980,CC1CC(C(N2CCN(C(=O)COc3ccc(Cl)cn3)CC2C)=O)CCC1C 23981,N1(C(c2cc(OCC)no2)=O)CC(C(=O)NC(c2ccccn2)C)C(F)C1 23982,c1(CC)nnc(CNC(c2cc(-c3cccnc3)on2)=O)s1 23983,C1(NC(COCCOC)=O)CC(NC(c2sccc2C#N)=O)C12CCC2 23984,C1(N(C)C(c2cccnc2S)=O)CN(C(=O)C=Cc2ccc[nH]2)CC1(C)C 23985,C(c1cccc(F)c1)=CCC(=O)NC(c1cn(CC(C(=O)OC)(F)F)nn1)C 23986,C1(C(=O)NC(C(=O)NCCCC)C)OCCOC1C 23987,CCS(=O)(=O)CC(=O)NC1(C)CC(NC(c2c(C(F)(F)F)coc2C(C)C)=O)C1 23988,c1(NS(C)=O)ccc(C2C(C(=O)NC(=O)CN(C)C(N)=O)C2)cc1 23989,Cc1c(CC(=O)NCC2CC2CNC(=O)CC2CCOCC2)cccc1[N+](=O)[O-] 23990,Cc1cccc(C(=O)NC2CCOCC2NC(c2oc(C(F)F)cc2C)=O)n1 23991,N1(C(CCCCN(C(=O)CCC2CCOC2)C)=O)CCn2nc(C)cc2C1 23992,C1(N)(CC)CCN(C(C2CC(=O)CCO2)=O)C1 23993,N1(C(C2(C=C)CCC2)=O)CC2C(NC(=O)CCCc3ccc(O)cc3)C2C1 23994,Cn1nnc2c1C(c1nc(-c3ccc(Cl)s3)nn1CC(F)F)CCC2 23995,Cn1cnc(C#N)c1C(=O)NC(c1cccc(Cl)c1)CNC(=O)CS(C)(=O)=O 23996,CCC(C)C(C(=O)NCCCC(C)(C)NC(C1C2CCC1CC2)=O)OC 23997,c1(C(N2CC=CC(NC(C3=CCN(C)C3)=O)C2)=O)nccc2occc12 23998,C(CC1CC1)(C(=O)NOC1CCC(O)C1O)NC(CC(COC)C)=O 23999,N1(C(C2C(C)N(C)CC2)=O)CCC2CN(C(=O)CNS(N)(=O)=O)C(C)C12 24000,c1(C(=O)NCC2N(C(CC#N)=O)CCOC2)cccc2c1OCC2 24001,C(C(=O)N1CC(NC(=O)Cc2c(F)cncc2Cl)CC(O)C1)(C(C)(C)C)SC 24002,c1(OC)cc(NCC2CN(C(c3cc(F)ccc3C)=O)CC2(C)C)nc(OC)n1 24003,c1(-c2c(OCC(F)F)ccnc2)ccc2c(c1)CN(Cc1cnc(O)c(Br)c1)C2 24004,C1(N(C(C2(CC)CCC2)=O)C)CN(C(=O)C=CCO)CCC1O 24005,C12(CC(=O)N(C)CC3CCC(CNC(C(=O)NCC)=O)CC3)CCC(CC1)OC2 24006,CCC(CC)C(C(=O)N1CCC(F)(F)C(CNC(C2C3CCCCC23)=O)C1)OC 24007,N1(c2n(CC3N(CC)CCC3)nnn2)CCS(=O)(=O)C(CC(=O)OC)C1 24008,c1(C(=O)NC2(C(=O)OC)CC23CCC3)cc(O)ccc1O 24009,c1(C(N2CC(CCNC(COC(C)(C)C)=O)C2)=O)c[nH]nc1-c1ccccn1 24010,c1(OC)ccc(C(=O)NC2CC(NC(=O)Cc3cscn3)C23CCC3)c(F)c1Cl 24011,O1NC(=O)C(CCC2CCC2)NC(=O)CCC1.C1(CC(=O)OC)CC1C1CC1 24012,C1(CCNC(C(C2CN(C(=O)C(C)(C)CO)C2)OC)=O)CCCCCC1 24013,c1(C(=O)NCC2C3CN(C(C4=CC(C)(C)C4)=O)CC32)[nH]cc2c1CCC2 24014,C(=O)(C(F)C(F)(F)F)N1C(CN(C)C(c2ccc(C(F)(F)F)s2)=O)COCC1 24015,c1(CCOC(c2cnn(CC)c2C(F)(F)F)=O)ccc(Br)cc1OC 24016,C1(C(=O)OC)CCCCN1C(C1CCCN1C(=O)CNC(c1ccnnc1)=O)=O 24017,C1(CC(c2nnnn2C2CCCCC2)(C)CCCNCCC(C)C)CCCC(=O)N1 24018,CCC(C)CCCCC(=O)N(C1CCCN(C(c2cnc(S)n2C)=O)C1)C 24019,Cn1ncc2c(NC3CC4CN(NC(C5C6CC7C(C6=O)C57)=O)CC34)ncnc12 24020,C(=O)(CCCCNC(c1ccn(C(F)F)n1)=O)NC(C=C)CO 24021,CCC(C)CC(C)C(=O)N(C)CC1CC(F)CN1C(=O)CCOC(C)CC(C)C 24022,CS(C)(=O)=Nc1ccc(C(N2CCN(C(c3ccc[nH]3)=O)C3CCC23)=O)s1 24023,C1(CC)(CC)CCCN1C(=O)CCc1cn(CC2(O)CCCCC2)nn1 24024,c1(C(N(CC(CN(C(C(C)=C(C)C)=O)C)O)C)=O)c(C)c[nH]c1CC(N)=O 24025,c1(-c2n(CCc3c(OC)nccc3)nc(C3CC3)n2)cc2c(OC)cccc2[nH]1 24026,C#CC1(O)CC(C(=O)NC(C)CN(C)C(c2cc(C3CCC3)[nH]n2)=O)C1 24027,Cc1cc(Cl)cnc1-c1cn(CCCC(=O)N(CC(C)(C)S(C)(=O)=O)C)nn1 24028,c1(OC)ccc(C2(C(=O)NCCCCNC(=O)CSC(C)C)CCC2)cn1 24029,C1(C(N2CC(C3(NC(C(c4ccnn4C)C)=O)CC3)C2)=O)CS(=O)(=O)CC(=O)N1 24030,N=c1cc(C(N2CCN(C(=O)C=CC3CCOC3)CC2CCO)=O)[nH]c(=N)[nH]1 24031,Cc1nc(-c2ncccn2)sc1C(=O)NCC1(NC(C2C3CCC23)=O)CCC1 24032,C1(NC(c2ccc(F)c(Cl)c2F)=O)CN(C(C2SCCS2)=O)CC12CCOCC2 24033,c1(CCC(=O)NC2CC(C)(NC(=O)C(O)C3CC3)C2)nnc(S)nc1O 24034,c1(OCC=C)ncccc1OC(c1nnn(C)n1)c1nnnn1CCCC 24035,c1(OCC)ccnc(C(N2CC(CCNC(C3(OC)CCOC3)=O)C(C)C2)=O)c1 24036,C1(NC(c2ccc(N(C)C)c(F)c2)=O)CN(C(C2(C)C=CCC2)=O)CC1C1CC1 24037,CCCC(CCC)C(=O)NCC12CCC(CN(C(=O)CCC(CC)CC)C1)C2 24038,C1(C(C(=O)N(C(COC)C)C)C)CCN(C(c2ccns2)=O)C1 24039,n1(CCCOC)c(N(CCC(=O)NC2CC2)C)nnc1-c1coc(C)n1 24040,c1(OCC(N2CCN(C(c3ccc(CO)cc3)=O)C3CC23)=O)ccc(Cl)c(F)c1 24041,c1(C(=O)NC(CC)(CNC(C2(C)CSC2)=O)CC)ccc2occc2c1 24042,c1(NC(C2C(NC(C(C(CC)O)(F)F)=O)COC2)=O)cnc2ccccc2c1 24043,N1(C(C(CCC)C)=O)CCN(C(c2cc(C(N)=O)c[nH]2)=O)C2CCC12 24044,C(=O)(C1=C(C)NC2=NCCCC2=C1)NCC1N(C(CC2CC(=C)C2)=O)CCCC1 24045,c1(C(N2CC3C(CC(=O)NCCC(CCC)C)C3C2)=O)ncc2ccccn12 24046,N1(C(C(Cc2ncn(C)c2)O)=O)CCCC2(CCN(C(=O)CNS(N)(=O)=O)C2)C1 24047,CP(C)(=O)c1cncc(CNC(=O)NC(c2ncccc2F)c2ccccc2)c1 24048,C#CCC(CC(=O)NC1(CC=C)CCOC1)NC(c1cnc(OC)cn1)=O 24049,C=CC(C)(C)CC(=O)NC12COC(C1)C(NC(C1CCCC1(F)F)=O)C2 24050,C(CCCC(=O)NCC(CO)OC)N(C(Cc1n(C)nnc1)=O)C 24051,c1(C(=O)NCC(CNC(C2=C(C)OCCS2)=O)CO)ccc2c(c1)OC(C)(C)C2 24052,C1(C(=O)OCC2CC(=O)N(C(=O)CCC3CCC3)C2)CCCN(C2CCCC2O)C1 24053,n1(CC(=O)NC2CN(C(c3ccc(NC(C)=O)nc3)=O)C2)c(C)cc(C)nc1=O 24054,c1(OCCNC(=O)C(c2ccc(I)cc2)F)c(F)cc(Cl)cc1F 24055,c1(C(=O)NCC2(OC)CCN(C(CS(CC)=O)=O)C2)cccc2c1OCC2C 24056,N1(C(C(C)Sc2ccccc2)=O)CCCC12CN(C(=O)C(c1ccccc1)O)C2 24057,N1(C(CC(C)SC)=O)CCCC(C)(NC(=O)C(=Cc2cnn(C)c2)C)C1 24058,C(=O)(CCC(=O)C(C)(C)C)NCC1C(C)CCCN1C(C1CCCCC1(C)C)=O 24059,c1(C(N2CC(CNC(c3c(CC)noc3)=O)C(O)C2)=O)c(S(C)(=O)=O)cnn1C 24060,C12COC(C)(C)CN1C2.c1(C(=O)NC2C(=C(C)C)CCCC2)ccc(O)c(F)c1 24061,N1(C(CCC(C)=O)=O)CCC2(CCCN2C(c2nn(C)c(C)c2Br)=O)CC1 24062,N1(C(CCNC(=O)NC)=O)CC(CO)CC1CNC(=O)CC1CCCC12CC2 24063,C1(CC(=O)NC(C#C)C(C)C)CCCCN1C(=O)C(C)NC(=O)CC 24064,C1(NC(c2cc(C)sc2C)=O)CC12CCN(C(c1nccnc1N)=O)C2 24065,N1(C(c2cccc(N)n2)=O)CCC2CC(CNC(=O)CCCCCO)CCC2C1 24066,N1(C(c2cnc(C)[nH]2)=O)CC2CC(NC(=O)Cc3csc(C(F)(F)F)n3)CC2C1 24067,C1(NC(c2c(SC)csc2)=O)CC2CCC1(NC(=O)CC(C)(C)C#N)C2 24068,C(=O)(C(C)CC(F)(F)F)NCCCCCNC(c1ccc(OCC(C)C)nc1)=O 24069,c1(CC(=O)NCCC(CNC(C(CC)C)=O)O)cccc2cnccc12 24070,CCCCC(C)(F)C(=O)NC(CC(=O)NCC(O)C1CCC1)C1CC1 24071,c1(NC(=O)CC2CC(O)CN2C(C2CCCSC2)=O)cc(O)cc(F)c1 24072,CC1CN(C(=O)CCF)CCC1NC(=O)CC1CCCNC(=O)C1 24073,Cc1c(NC2CC(C)NC(C)C2)ncnc1N(C)CC1CCOCC1 24074,N1(C(c2n(C)c(Cl)c(Cl)c2)=O)CCC2(CCCCC2NC(=O)Cc2cnc[nH]2)C1 24075,CCC(CC(=O)NC1CCC(C)N(C(c2nc(C)sc2C)=O)C1)CC(C)C 24076,c1(C(=O)NCC(CNC(c2cc(C)ccc2N)=O)OC)coc2c(Cl)cccc12 24077,c1(C(COC(C(C)C(C)S(C)(=O)=O)=O)=O)c(Cl)cc(Cl)cc1C#N 24078,N1(C(CCC2(C)CCC(=O)N2)=O)CC2CCC(C1)C(NC(=O)CC1CC1)C2 24079,C12(C(=O)NC(CCOC)CNC(c3ccsc3SC)=O)CCC(OC)C1C2 24080,C1(CNC(C2CC(CNC(=O)C(C3CCOCC3)F)C2)=O)CC2CCCC2C1 24081,Cc1ccc2c(C(=O)N(C3C4CN(C(C5CCC(C)CC5)=O)CC34)C)onc2c1 24082,C=CCCC(C(=O)NCCC(O)C(F)F)NC(=O)C(=O)NC1CC1 24083,c1(C(=O)NC2C(NC(CC3(C=C)CCC3)=O)CCCC2)cc(F)c2[nH]nnc2c1 24084,c1(OC)cc(C(N2CCCC2CNC(C2C(C#N)C2(C)C)=O)=O)cc(Cl)c1 24085,c1(C(N2C(CNC(C(C)CC(N)=O)=O)(CO)CCC2)=O)cnn2cccnc12 24086,c1(C(N2CC(N3CCN(C(C4CC4(F)F)=O)CC3)C2)=O)n[nH]c2ccc(Cl)cc12 24087,Cc1ncc(C=CC(N2CC(F)(F)CC2CCNC(=O)C(C)C(F)F)=O)c(O)n1 24088,c1(C(=O)NCC(CNC(c2sc(CC)c(C)c2)=O)CO)ccc2cccnn12 24089,C1(NC(=O)OC(C)(C)C)C2CC3CN(C(=O)NC4CCCCO4)C1C3C2 24090,c1(COC)nc(CC(=O)NCC2CC2N)cs1.C1(=O)CC12CC2.CSC 24091,C1(CNC(C(C)C(F)F)=O)CCC2(CC1)CCN(C(=O)CC1CC13CC3)CC2 24092,C#CC1CN(C(C2(NC(c3cnc(Cl)n3C)=O)CCCC2)=O)CCN1C 24093,N1(C(CC(=C)C)=O)CCC(N(CCO)C(C2CC(=C3CC3)C2)=O)CC1 24094,Cc1ccc(C=CC(=O)NCCCC2CCCN2C(=O)CN(C)C)nc1 24095,C1(CCC(=O)N(C(C=C)C)C)CCCCN(C(c2cc(=N)[nH][nH]2)=O)C1 24096,C(=O)(CCC(C(C)C)NC(c1ccncn1)=O)N1CCC(C(CC)C)CC1 24097,c1(N(CCNc2cccc(C)n2)C)nc(=NCCn2ncnn2)[nH]c2c1CCC2 24098,C(CC(COC)N=c1[nH]c(=NCC2(N(C)C)CCSC2)[nH]c2c1SCC2)OC 24099,N1(C(C(CC#C)O)=O)CC2CCCC(C1)N2C(=O)CN1CCCC(CC)C1 24100,CC(C)(C#N)C(=O)NCCc1ocnc1CNC(=O)CCc1nncs1 24101,C1(COc2cccc(NC(C3CC(S(C)(=O)=O)C3)=O)c2)CC2(CCOCC2)CO1 24102,N1(C(C2CC(C)(C(=O)OC)C2)=O)CC(NC(=O)Cc2cc(C)on2)C(O)C1 24103,CC1C(NC(C2(CCO)CC2)=O)CC2CCC1N2C(c1c[nH]nc1C(C)(C)C)=O 24104,c1(C(N(C2CCN(C(=O)OC)C2)CC)=O)ccc(NC(=O)CC2(C)CCCO2)cc1 24105,C(=O)(C(C)CC(C)(C)C)N(C(C)C(=O)NCCCC(N)=O)CC 24106,C1(NC(C2(CC=C)CC2)=O)CS(=O)(=O)C2CN(C(C3CC(OC)C3)=O)CC12 24107,N1(C(CCC=C=C)=O)CC2(C1)CN(C(c1cc(C)nc(C)n1)=O)C2 24108,c1(OCC)ccc(C2CN(C(=O)C3CC3)CC2NC(C2CC23CC(O)C3)=O)cc1 24109,C1(C(N2CCCC(C3N(C(c4c(C)noc4C)=O)CCC3)C2)=O)CC(C2CC2)=NO1 24110,C12(CNC(c3c(C)cccc3)=O)CCCC1CCN2C(=O)Cc1cnn(C)c1C 24111,c1(OC)cc(OC)cc(CN2CCC(O)C(C(=O)Nc3ccc(C)cc3C)C2)c1 24112,C1(C(=O)NCC2(C)N=C(C)SC2)CC(C)(C)CN1C(=O)CCC1CCCCC1 24113,c1(C(CC)C)ccc(C#N)c(NC(Cc2nccn2C)C(C)C)n1 24114,C(=O)(C(C#N)C(C)C)NCC1(C(=O)NCCc2ncc[nH]2)CC(=C)C1 24115,C1(CC=C)(C(N2CCC(n3cccn3)C2)=O)CN(C(=O)C(O)CN2CCCC2)C1 24116,Cc1nc2sccn2c1C(=O)NC1CN(C(c2cccc3oncc23)=O)C1 24117,C1(CNC(C2CC(SC)C2)=O)CN(C(C2CCN(C)C2=O)=O)CC1(F)F 24118,C(=O)(C1=Cc2cccc(OCC)c2OC1)NCC(CNC(CCC)=O)O 24119,C(CC(O)C(=O)NC1CC(NC(=O)CCSc2ccccc2)C1)SC 24120,c1(CC(=O)NCCOCCN(C(=O)C(O)CF)C)ccccc1OC(F)F 24121,c1(N(CCCC(F)(F)F)C)nc2c(c(=NCCc3n[nH]c(C4CC4)n3)[nH]1)CCC2 24122,c1(COC(C2CC(=C(F)F)C2)=O)cccc2ncccc12 24123,C1(NC(c2c(SC)n(C)nc2)=O)COC2(CCN(C(=O)CC3CN(C)C3)C2)C1 24124,c1(C(=O)NCC(COC)O)n[nH]cc1CNC(=O)CN1CCCC1C 24125,C1(C)(C(=O)NCC(CC)NC(=O)C(N2CCCCCC2)C)CC(C2CC2)=NO1 24126,c1(C(N2CCC(O)(CN(C(C3C(OCC)C3)=O)C)C2)=O)cnc2cnccc2c1 24127,C(=O)(N1CC(O)CCO1)C1(CC)CCN(C(=O)C(O)CC(F)(F)F)CC1 24128,C1(C)(C(=O)NC(CNC(c2cc(CC)c(CC)o2)=O)C)CCC2(CC1)OCCO2 24129,C1(C)(C(N(C)CC2(CNC(c3cc(CC)oc3C)=O)CC2)=O)CC(C(C)C)=NO1 24130,C1(NC(c2cccnn2)=O)CC(F)CN(Cc2cc(B(O)O)co2)C1 24131,CC1CCCC(CCNC(=O)CC2CC(O)CN2C(c2cnn(CCF)c2)=O)C1 24132,N1(C(CCCCOC)=O)CC(CNC(=O)C2=NOC(C(C)(C)C)C2)C(F)(F)C1 24133,N1(C(C(CCCCC)C)=O)CCCC2(CCCN2C(c2cccnc2C)=O)CC1 24134,Cc1nn(-c2ccccc2)cc1C(=O)NCC1C2CN(CC(O)C(F)(F)F)CC12 24135,Cc1cc(C)c(CC(=O)NCC(F)CNC(=O)C(c2ccccc2)=O)s1 24136,C(CC(O)C(=O)N1CC=CC1CNC(=O)CSC(C)C)SC 24137,C12(NC(C(CCC)O)=O)CCC(CC1NC(=O)CN1CCN(C)CC1)C2 24138,n1(CC)nnc(C(=O)NCc2csc(CNC(c3cc[nH]n3)=O)n2)c1C 24139,c1(C(=O)NC2C(NC(CC3CC(=O)NC3)=O)CCC2)cccc2nccnc12 24140,Cc1nc(C2CC2)ncc1C(=O)NC(CCNC(=O)C(C)NS(C)(=O)=O)C(C)C 24141,CC(C)(C)CCCC(=O)NC1CCN(C(=O)CC2(CCCO)CCCC2)C1 24142,c1(CNC2(c3n(CCCF)nnn3)COC3(CCC3)C2)nc2c(s1)CCCCC2 24143,CC1CCCN(C(c2csc(CO)n2)=O)C1CO.C12(CCOCC1)C(=O)N2 24144,N1(C(C2(F)CCC2)=O)CCC2CN(C(=O)C(F)(F)Cl)CC2C1 24145,Cc1cc(O)c(F)cc1NC(C1CCN(C(c2cscc2Cl)=O)C1C(C)C)=O 24146,N1(C(CCCC=C)=O)CC(C(N2CCCC2CSC)=O)C2(CC2)C1 24147,CC(CCCCNC(c1cnnn1C)=O)NC(=O)CCn1ncn(C)c1=O 24148,N1(C(CNC(C)=O)=O)CC(C(N)=O)(CNC(C2(c3ccno3)CCC2)=O)C1 24149,Cc1coc(C)c1C=CC(N1CC(O)(CCNC(C2COC(C)C2)=O)C1)=O 24150,C1(N(C(C=CC)=O)C)CN(C(=O)C(C)N(CC(F)(F)F)C)CC1(C)C 24151,c1(C(N(CC(O)CO)CC)=O)cnn(CCNC(c2nscc2C)=O)c1 24152,c1(CC)[nH]nc(C(=O)NCCC2(OC)CN(C(=O)C(C)OCCO)C2)c1[N+](=O)[O-] 24153,C1(C(N(C2CCN(C(=O)OC(C)(C)C)CC2)C2CC2)=O)SC2C=CC1CC2 24154,CC(C)C(C)CC(=O)NCC1CCCCN1C(c1cccc(-n2cncn2)n1)=O 24155,C1(NCCN2CCC(C(=O)NC(c3ccc(Cl)s3)C)C2)CC2(CC(=O)C2)C1 24156,Cc1c(C(N2CCN(C(c3c(Cl)cnn3C)=O)C3CC23)=O)cccc1O 24157,c1(COC)ccc(C(=O)NCC2CC(CNC(=O)CCc3cncn3C)CO2)o1 24158,N1(C(C(C=CC)O)=O)CCCN(C(=O)Cc2ccc(Br)cc2OC)CC1C 24159,c1(C(=O)NCC2(Cn3cc(C(C4CCCC4)OC)nn3)CC2)nnc(O)nc1O 24160,C1(=O)CC(c2ccccc2)N1.C1(CN)CCCN1C(=O)CCCN1CCCC1 24161,S(=O)(=O)(c1cnc(NC(C)Cc2cccc(C)c2)cc1C)NCCN(CC)CC 24162,C1(C)(C(=O)NCCCNC(C2(C)CC(C(F)(F)F)C2)=O)CC2CC2C1 24163,C(=O)(C(O)CC(F)F)N1CC(O)(CCNC(CCC2C(C)=NOC2=O)=O)C1 24164,C1(CC)CCCCC1NC(C1(CC)CN(C(=O)COCC2CCCO2)C1)=O 24165,C1(CC(N2CC(C)C(NC(c3cnc(O)c(F)c3)=O)C2)=O)CC2(CCCC2)CO1 24166,N1(C(CCC(=O)N2CCC(O)CC2)=O)CC2(C1)CN(C(=O)CN1CC3CC3C1)C2 24167,c1(C(=O)NC(C)CCCNC(C2CC3CC3CC2C)=O)ccc(F)c2c1CCC2 24168,c1(C(=O)OCC)c[nH]c(=NCC2CCCCN(C(=O)CCc3nc[nH]n3)C2)s1 24169,C1(C(=O)NC2C(C)N(C(c3cc(Cl)cc(Cl)c3N)=O)CC2)OCC2COCCC12 24170,N1(C(COCCOCC#C)=O)CCCC12CCCN(C(=O)C=CC)C2 24171,CC1(C)C2CCC(C2)C1(C)C(=O)NCc1ccccc1CNC(c1csnn1)=O 24172,C1(C(=O)NCC2(F)CN(C(Cn3cc(C(=O)NC)nn3)=O)C2)C2CC3C(C2=O)C13 24173,c1(CC(=O)NCC(C)NC(=O)CC2CCCC2)ccc2c(c1)CC2 24174,c1(C(=O)NCCCNC(C=CCOC)=O)cc(C)ccc1S(N)(=O)=O 24175,c1(N2CCC(NC(=O)NC(COC)C(=O)NC(C)(C)C)C2=O)ccncc1N=[N+]=[N-] 24176,c1(CC(N2C(C(C)(C)NC(C3CC4C=CC3C4)=O)CCC2)=O)cccc(Cl)c1Cl 24177,N1(C(C2(CC)COC2)=O)CCC(C2CCCN(C(=O)C=CCO)C2)CC1 24178,N1(C(c2c(C#C)c[nH]n2)=O)CCC(C2CC2)C1CNC(C1C=C(C)CS1)=O 24179,CC1CN=C(NC(C2CCCN2C(=O)OCc2ccccc2)=O)S1 24180,c1(C(C)C)ccc(C=CC(=O)NC23CCC2CN(C(=O)CC2CC(F)C2)C3)cc1 24181,Cc1nc2cnn(C)c2cc1-c1ccc(C2CCC(C#N)(C(=O)O)CC2)cc1 24182,c1(C(=O)NCCC(CNC(c2ccnn(C)c2=O)=O)O)c2c(nn1C)CCSC2 24183,CC1CC(NC(C2CN(C)C(=O)N2)=O)CCN1C(=O)Cc1nnc(O)s1 24184,c1(CC(=O)NC2CCOCC2NC(=O)CC2CCOC2)ccccc1F 24185,C1(O)(NC(N2CC(NC(C(C)NC(c3ccccc3)=O)=O)C2)=O)CC2CCC1C2 24186,C(=O)(C1=C(C#N)CCC1)NC(CC(=C)Cl)C(=O)N1CCCC(F)(CO)C1 24187,c1(C(N2CCCC(CNC(C3C(CC)CCO3)=O)C2)=O)cc2cc[nH]c(=O)c2s1 24188,C1(C(=O)NC2(C(=O)NCC3(OC)CCCC3)CC2C)CCC(=O)NC1 24189,c1(C(N2CC(C(=O)NCC(CCC)OCC)(CC)C2)=O)cc(C)ccc1F 24190,C1(C(=O)NCC2(F)CCN(C(C(c3cccnc3)C)=O)C2)Cc2cscc2C1 24191,CCC(CC(=O)NC(C)(CO)C(=O)NC1(CC(=O)OC)CC1)SC 24192,c1(CC(=O)NC2CCCCC2NC(c2ocnc2CC2CC2)=O)ccc(O)cc1 24193,C12(C(=O)NC3CCC(NC(COC)=O)CC3)CCC(C1)C(C)(C)O2 24194,C(=O)(CCCCCF)NCc1c(C(=O)NCC2(OCC)CCOC2)nco1 24195,C1(C(=O)OCc2nnc(C)o2)CC(F)(F)CS1 24196,C1(C)(C(=O)NCCCOCC)CCCN(C(=O)CC2CCOCC2)C1 24197,C1(C(COC(C2CCN(CC(=O)Cc3ccccc3)C2)=O)=O)CC2CCC1C2 24198,CC1(C)CCCC1CCNC(=O)C(=O)Nc1ccc(CN2CCCCC2)cc1 24199,S(=O)(=O)(c1ccc(N(C(C)CCC(C)C)C)cc1Br)NC(c1scc(CC)n1)C 24200,O=S1CCC(N=c2nc3sccc3c(NCC3(n4ccnn4)CC3)[nH]2)C1 24201,C(=O)(CCS(N)(=O)=O)NCC(CCNC(=O)C(c1cccc(C)c1)F)OC 24202,N1(C(C(COCC)N=[N+]=[N-])=O)CCC2CN(C(C3CC3C(=O)OCC)=O)CC2CC1 24203,Cc1ccn2cc(C(N3CCC(C)CC3CNC(=O)CC3CCCO3)=O)nc2c1 24204,c1(N(C)Cc2ccc(Cl)s2)[nH]c(=NCc2cc(N)ccc2F)nc2scnc12 24205,CCC(C)(CO)C(=O)NC1CCCC1NC(=O)COC1CCCCCC1 24206,N1(C(C(CC)OC)=O)CCN(C(C2CCC(C)(OC)CC2)=O)C2(CCC2)C1 24207,N1(C(C(C)OCC#C)=O)Cc2nccn2CC(NC(=O)C2=CCC(C)(C)C2)C1 24208,c1(C(=O)NC(CCC)C)cccc(-n2cc(-c3cnccn3)nn2)c1 24209,N1(CCC)CCCC(C(=O)NCCC2CN(C(c3ccc(C)nc3)=O)CCO2)C1 24210,c1(CC)cc(C(=O)NC(C2(O)CCN(C(C3(OC)CCOCC3)=O)C2)C)sc1C 24211,C(=O)(CCC(C(=O)NCC1CCN(C(=O)C(O)C(C)(C)C)CC1)N(C)C)OC 24212,c1(NC(=O)NC(COC(F)F)C2CC2)ccc(N=Nc2ccc(O)cc2)cc1 24213,CC1CN(C(c2ccc(C(C)(C)C)cc2N)=O)CCC1NC(c1csnc1Cl)=O 24214,C1(C(=O)NC2CCC(NC(CC3(COC)CCCC3)=O)CC2)OCC2CCCC12 24215,c1(NC(C2CC2C(=O)NC2C3COCC23)=O)ncc(Cl)nc1Cl 24216,N1(C(=O)CCCF)CCCC2C1CCCN2C(c1cc2cccnc2s1)=O 24217,C1(C(=O)NCCN(CCC)C(C2(CCC)CC2)=O)CCn2cnnc2C1 24218,c1(C(=O)NC2C(NC(C3CCC(C(=O)OC)CC3)=O)CC2)cc(SC)cc(F)c1 24219,C1(C)(CNC(C2C(OC)C2)=O)CN(C(c2ccc(Cn3ccnn3)o2)=O)CCO1 24220,c1(CNC(N2CCC(c3ccncn3)C2)=O)cc(O)ccc1F 24221,N1(C(c2c(OC)c[nH]n2)=O)CC2OCCN(C(C3CC34CCSCC4)=O)C2C1 24222,C1(N(C(=O)CC2CC23CC3)CC)CCN(C(=O)CC2OCCO2)CC1 24223,c1(CNC(C(COC)OC)=O)ccc(CC(C)NC(c2c[nH]c(C#N)c2)=O)cc1 24224,C(=O)(C(O)Cc1cnc[nH]1)NCC(C1CC1)NC(C1(OC(C)C)CCC1)=O 24225,C12(NC(=O)Cc3cc[nH]n3)CC(CNC(C3(N4CCOCC4)CCCC3)=O)(C1)C2 24226,CC1CCn2cc(C(N3CCCNC(=O)C3c3ccccc3)=O)nc2C1 24227,c1(C(=O)NC(CCOC)CNC(C2(C)CCCCC2)=O)cc(=O)n2nccc2[nH]1 24228,N1(C(CCC)=O)CCCC(CO)(NC(c2nn(C)cc2SCC)=O)C1 24229,C=CC(C)(C)CCN=C(NCC(Br)=CCC)NC1CCN(C(=O)OCC)C1 24230,c1(CCNC(C2CCCN2C(=O)CCc2ccncn2)=O)cc(CO)ccn1 24231,C12CCCN(C1)C(=O)CNC(=O)C(N(C)C)CNC(=O)N2.C(C)(C)(C)NC(N)=O 24232,Cc1ccccc1C(C)(C)CNC1CCOC(c2ccc(F)cc2)C1 24233,c1(C2(C(=O)NC(C)CC3CN(C(=O)CC4CSC4)C3)CC2)ccncc1 24234,C(CC(O)CC(=O)N1CCCC1CN(C)C(c1cnccn1)=O)SC 24235,C1(CNC(C=Cc2n(CC)ncc2)=O)CCC12CCN(C(=O)C(F)OC)CC2 24236,CCCCC(C)CCC(=O)NC1(COC)CN(C(=O)C(C)CN(C)C)C1 24237,c1(C(=O)NC2(CNC(c3cc(Br)no3)=O)CC2)ccc2c(c1)CCC2=O 24238,Cc1cc(C(=O)NCC2(NC(=O)C(C)OCCC(C)C)CCC2)c(O)c(C)n1 24239,c1(CCC(=O)NC2CN(C(c3c(C)n[nH]c3)=O)C(C)CC2)n[nH]c2c1CCCC2 24240,CS(=O)(=O)CCC(=O)NC1C2CC1CN(C(=O)CCc1cccc(O)n1)C2 24241,S(=O)(=O)(c1cc(Br)ccc1Br)N(C)CC1CN(C(c2ccnc(Cl)c2F)=O)C1 24242,c1(C(c2n(CCOC)nnn2)NCC2(OCC)CCOCC2)cncc(F)c1 24243,C(=O)(CC1=CCN(C(=O)CCC(=O)NCC)CC1)NC(CCCC)C(=O)OC 24244,C1(NC(c2cn(CCC)nc2)=O)(CO)CCN(C(c2cccc(O)n2)=O)C1 24245,O=C1NCCC2CCN(C(c3cc4occc4s3)C(=O)NCc3ccco3)C12 24246,c1(-n2cc(CC3(C(=O)O)CCCCO3)nn2)cccc2c1OCO2 24247,c1(OC)cc(F)c(COC(C2CCC2c2ccc(Cl)c(Cl)c2)=O)cc1OC 24248,c1(OC)ccc(C(=O)NC2CC(NC(c3ccn(CCSC)n3)=O)C2)c(F)c1F 24249,C1(C(=O)NC2C(CC(=O)NC(C3(CO)CCC3)C)C(O)C2)CC2C=CC1O2 24250,Cc1c(C(=O)NC(C2CCCN2C(=O)Cn2cnc(=N)[nH]2)(C)C)ccn1C1CC1 24251,C1(COC)(CNC(=O)Cc2coc(C)n2)CCN(C(=O)C(C)(C)C2CCC2)CC1 24252,N1(CC)CCC(C(=O)N(C)CC=CC(=O)NC2CC2C)C1 24253,n1(CC)ncn(NC(=O)Cn2cc(C(C)NC(C34CC(CO3)C4)C)nn2)c1=O 24254,C1(NC(C(=O)NCCOC)=O)CC2(C1)CC2C(=O)Nc1ccccc1C(C)(C)C 24255,c1(COC(C2CN(C(C3CC3(c3ccccc3)F)=O)C2)=O)csc(C(F)(F)F)n1 24256,C1(c2ccc(OC)cc2)CC(C(=O)NCCCC2CC(C)(C)CO2)=NO1 24257,C1(NC(C(C)CS(C)(=O)=O)=O)COC2(CCN(C(C3C4(CC4)C34CC4)=O)CC2)C1 24258,C1(OCC(N2CC(C(C)NC(C(C3CCC3)OC)=O)C2)=O)CCC(C)CC1 24259,C(=O)(CCCCC(=O)NCC1(CCNC(C2CCC(F)C2)=O)CC1)OC 24260,C(=O)(CCCCCNC(C)=O)NCC1CN(C(c2n(CC)nc(C)c2)=O)C(C)C1 24261,c1(OC)cc(F)ccc1C(=O)NC(CNC(C1CC=C(C)CC1)=O)C1CC1 24262,C1(C(=O)OC)CCN(C(=O)C2CN(C(=O)CN3CC4CCC3C4)CC23CC3)O1 24263,C1(CNC(=O)CCc2nc[nH]n2)COC(CNC(C2CC(O)C2)=O)C1 24264,N(C(=NCCCCl)NCC1CC12CCCC2)Cc1ccc(OC)cc1 24265,C1(CC(=O)NCC2CCN2C(=O)CC2CCC(O)C2)CN2CCC1CC2 24266,C(C(=O)OC)(C(C)(O)C(F)(F)F)NCc1c(CC)ccc(F)c1 24267,c1(NC(CN(CCC)CCNC(=O)CNS(=O)(=O)CC)=O)nc(C)nn1C 24268,C1(OC)(CNC(=O)CCc2ncnn2C)CN(C(c2ccc(C(C)C)s2)=O)C1 24269,c1(OC)c(Cl)nc(NC(c2csc(NC(c3nc(Br)ccc3F)=O)n2)=O)nc1Cl 24270,C1(CNC(c2c(OC)cccc2)=O)CCCCN(C(c2c[nH]c(=N)nc2O)=O)C1 24271,c1(-n2cc(C(C)NC(c3c(C(=O)NC)occ3)=O)nn2)ccccc1CC 24272,c1(C(=O)NC2C(N(C(COCCC)=O)C)CCCC2)cc(C)c(O)c(N)c1 24273,N1(C(c2c(N)non2)=O)CCC(NC(c2ccn(C3CC3(F)F)n2)=O)C(CO)C1 24274,C(=O)(C(F)C(C)(F)F)N1CC(C)(OCC(=O)N(C)CC2CC2(F)F)C1 24275,C(C1=CCN(C(c2ccc(Br)cc2F)=O)CC1)NC(C1CC12CCCC2)=O 24276,C(=O)(CC(C)C(F)F)NCCCCC1CCN(C(C2(CC)CC(F)(F)C2)=O)CC1 24277,c1(OC)nccc(Br)c1C(=O)NC1CC(N(C)C(C2CN(C)C(=O)N2)=O)C1 24278,c1(C(=O)NC2CC(N(C(c3cnc(OCC)s3)=O)C)C2)nccc(OC)c1N 24279,CC(C)C(C)(O)C(=O)NC(c1ccccc1)CNC(c1ccns1)=O 24280,c1(C(CC)NCC2CCC(C)O2)ccc(O)c(Br)c1 24281,c1(C(N(CCC)CCNC(=O)C(C)C2CCOC2)=O)c(F)ccc2nc[nH]c12 24282,C(CC(C(C)C)(c1nnnn1C(c1ccccc1)C)Nc1ccc(O)cc1)OC 24283,C(CCC(=O)N1CC(C(N)=O)C1)(C(C)C)NC(C=Cc1cc(C)no1)=O 24284,c1(C(=O)NCCC2(C)CCN(C(=O)CCC3CC3)C2)ccn2ccnc2c1 24285,Cc1cc(C(=O)NCC2(CNC(=O)C=Cc3cncs3)CC2(F)F)ccc1O 24286,CC1C2CC(C2NC(C2CCC(F)(F)CC2)=O)N1C(c1c[nH]c(=O)cn1)=O 24287,C1(CC)CN(C(=O)C(C2CCCCC2)O)CCN1C(c1cc(C)n(C)c1)=O 24288,N1(C(C(CC)OC)=O)CCN(C(c2cc(S(C)(=O)=O)co2)=O)C2CCC12 24289,C1(C(N2CC(C)C(N=[N+]=[N-])C2)=O)CC(F)(F)C12CCCC2 24290,c1(C(=O)NC2C3(CC(NC(=O)COCC(F)F)C3)C2)ccc2cnnn2c1 24291,C1(NC(C2CCCC(NC(CC3(C#N)CC3)=O)C2)=O)CC2(CNC(=O)O2)C1 24292,CC1CCN(C(=O)CCc2c(F)cccc2F)CC1NC(=O)C=C1CCCCC1 24293,N1(CC(=O)NCC2(O)CN(C(c3c(N)cc(Cl)nc3)=O)C2)CCCCCCC1=O 24294,C1(NC(c2c(Cl)cn(CC)n2)=O)COCCN(C(=O)C(C)Cn2ccnc2)C1 24295,c1(C(=O)NC(C(=O)NC(CCOCC)C)c2cccs2)cc2ccccc2o1 24296,C(C)(C(=O)NCC1CC([SH](CCC(=O)NCC(N)=O)C)C1)OCCOCC 24297,N1(C(C2CC(=C)C2)=O)CCC(CF)(NC(c2cnc(C3OCCO3)s2)=O)C1 24298,c1(N2CC(C)(C)S(=O)CC2)nc(N2CC3OC(=O)OC3C2)nc2c1SCC2 24299,C1(CC)CCCCC1C(N1CCC1(C)C)C(=O)Nc1ccccc1Cl 24300,c1(CNC(C2C(C)C2)=O)ccc(CN(C)C(C2CCC2C(=O)OC)=O)cc1 24301,Cc1c(CC(=O)NCC2(CCNC(=O)CC3CC=CC3)CC2)ncn1C 24302,N1(C(CNS(C)(=O)=O)=O)CC2COCCC2(NC(c2ccn3cncc3c2)=O)C1 24303,Cc1cccc(C(=O)N(C2CCC(NC(C3CN(C)CCO3)=O)CC2)C)n1 24304,N12CCC3(CCC(O3)C1=O)CC2.c1(C(C)=O)ccccc1C(=O)NC(C)(CO)CO 24305,c1(NC(COC(C)(C)C)CO)ccc(S(=O)(=O)NCC2CC2(Cl)Cl)cc1Br 24306,C1(C(N2CCC(OCCNC(C(C=C)O)=O)C2)=O)CCC2C(CC1)C2(F)F 24307,N1(C(c2c(C)ccs2)=O)CCC(NC(=O)C(c2ccc(F)cc2F)C)C(F)C1 24308,C=CC(CC(=O)NC(C1CCN(C(=O)CC(F)(F)F)CC1)(C)C)c1ccccc1 24309,C(=O)(C1=C(C#N)CCC1)N(C1CCN(C(=O)C(c2cccnc2)OC)CC1)CC 24310,c1(OCC=C)ccc(Cl)nc1C(=O)NC1CCCCC1NC(=O)C(O)C(C)(C)C 24311,c1(CC(=O)NC2CC2CNC(C2CS(=O)(=O)C2)=O)cc(F)c(F)cc1F 24312,C(C(C)C(F)C(=O)N1CC(OCC(F)F)C1)NC(c1cc(CCC)[nH]n1)=O 24313,C1(C(=O)NCC2(C)CCN(C(c3nccc(CC)c3)=O)C2)CCCCS1(=O)=O 24314,c1(C(=O)OC)cnc(NCC2CC(C)N(C(=O)CN(S(C)(=O)=O)C)C2)nc1 24315,c1(C(C(N2CCC(O)(C(C)C)C2)=O)(F)F)ccc2c(c1)OCO2 24316,Cc1cncc(C(=O)NCC2CC2CNC(c2ccc(=N)[nH]c2Cl)=O)c1Cl 24317,N1(C(c2cc(C)nn2C)=O)CCN(C(c2c(C)coc2C)=O)CC12CC2 24318,c1(OC)ccc2nc(N3CC(NC(C4(C)COC4)=O)C(C)(C)C3)sc2n1 24319,N1(C(c2cccn(C3CCSC3)c2=O)=O)CCS(=O)(=O)N2CCCC12 24320,Cc1cc(C)nc(SCC(=O)N(C2CCCN(C(=O)C(C)C(C)(C)C)C2)C)n1 24321,Cc1ccc(Br)c(F)c1C(N1CC2CC1C2C(N1CC2CC1CC2(F)F)=O)=O 24322,C(=O)(CC(O)C(C)C)NC(CCOC)C(=O)NC12CC1CN(C)C2 24323,N1(C(CN(C(=O)C(O)C(C)CC)CCC)=O)CC2(COCC(=O)N2)C1 24324,c1(C(N2C(CNC(C3CCCC(C)(C)C3)=O)COCC2)=O)cnn2c1CCCC2 24325,N1(C(=O)NCc2c(CC)ccc(F)c2)CCc2cc(OC)ccc2C1C 24326,c1(COC)nc(OC)cc(NCC2CCCCN(C(c3conc3C)=O)C2)n1 24327,c1(SCC(=O)NCC2CC2CNC(c2cccnc2C(F)F)=O)ccc(O)cc1 24328,C(C(=O)N1CC(NC(=O)CC2(CO)CCC2)C(C)C1)(C(C)(C)C)NC(C)=O 24329,c1(C(=O)NC2(CNC(=O)CC3CCCS3(=O)=O)CCCC2)cccc2nsnc12 24330,C1(C(=O)NCCCN(C(C(C)SCC)=O)CCO)CCCC1n1ccnn1 24331,C(C(CC(C)C)C(=O)N(C)Cc1c(C)cnn1C)NC(CC(C=C)C)=O 24332,C1(NC(C(CC)N(CC)CC)=O)COCCC1NC(c1cnc(C2CC2)s1)=O 24333,N1(C(C(CC)C)=O)CCN(C(=O)CNC(c2ccccc2C)=O)CC1 24334,c1(CC)cccc(C(=O)N(C)CC2CCCN(C(=O)C(C)N(C)C(C)=O)C2)c1N 24335,c1(OC(CC(CC)N(C)CCOC)=O)ccccc1C#N 24336,C1(C(=O)NCC(C2CCOCC2)CC)CCC(C2CCC2)CC1 24337,c1(CC)ccc(C(=O)NCCC2(C)CCN(C(c3ocnc3C3CC3)=O)C2)cc1 24338,N1(C(c2c(OC)nsc2)=O)CC2CC(NC(=O)C(C)CCO)C2C1 24339,c1(C(=O)NC2CCC(CNC(C3(COC)CC(=C)C3)=O)C2)c(F)cc(Cl)cc1F 24340,N1(C(c2n(CC)ncc2)=O)CC2(CC2)CC1C(N1CCC(N2CCC2)C1)=O 24341,C(=O)(CCCCCN=[N+]=[N-])N1CC(CC)N(C(=O)CC(C)c2cnn(C)c2)CC1 24342,CCC(C)C(O)CC(=O)NCCCC(CO)NC(=O)CCCn1ccnc1 24343,c1(C(=O)NCC(CN(C(C(C)SCC)=O)C)O)ccn(CCN(C)C)n1 24344,c1(C(C)C)cccc(C(=O)NC2CC(NC(=O)CC3CCC(C)(C)C3)CC2O)c1 24345,N1(C(c2c(SC)snn2)=O)CC(NC(C2(C(C)(C)C)CCCCC2)=O)C(C)C1 24346,c1(C(=O)NC2(C3CN(C(CS(C(C)C)(=O)=O)=O)C3)CC2)cc2cc(Cl)cnc2o1 24347,CC1(C)CCCOC1CC(N1CCOC(CNC(C2CC(=O)N(O)C2)=O)C1)=O 24348,N1(C(C(C2CCC2)OC)=O)CC(CNC(C2CCCCC2O)=O)C(C)C1 24349,Cc1cc(C(N2CCC(CNC(c3ncccc3C)=O)C(C)C2)=O)[nH]c1C#N 24350,C1(C(N2CCC(N(C(C(c3ccccc3F)C)=O)CCO)C2)=O)C(C)(C)C1(F)F 24351,Nc1ccc(C(=O)NC2CCOC(C3CCN(C(C4(F)CCC4)=O)CC3)C2)cc1 24352,Cc1ccc(S(=O)(=O)N2CCN(CC(=O)NC3CCCC3)CC2)nc1 24353,Cc1ncnc(C(N2CC3CC3(CNC(c3cn(C)c(O)n3)=O)C2)=O)c1C 24354,C=CC1CCCCN1C(=O)Cn1cc(CNC(=O)COCC2CC2)nn1 24355,c1(COC(C(=O)NC2CCC(CCNC(C=CCC)=O)C2)C)ccc(C)cc1 24356,c1(C(N(C(C)C(=O)NC2CCOCC2OC)CC)=O)cnn2ccccc12 24357,N1(C(c2c(CC)con2)=O)CC(NC(C2CCC(C(F)(F)F)CC2)=O)C2(CC2)C1 24358,c1(N2CC(OC)C(F)C2)nc(Nc2cc(N)ccc2C)c2cnn(C)c2n1 24359,n1(CC)cc(C(=O)NCCC2(NC(=O)CC3CCNC3=O)CCC2)c(C)n1 24360,Cc1ccc2c(C(=O)NC3CCN(C(=O)C#CC4CC4)C(C)C3)n[nH]c2c1 24361,c1(N(CCNC(C2(C(=O)OCC)CC2)=O)C(=O)CC)ccc(C)cc1.C12CC1N2 24362,c1(C(=O)NCCC2CC(NC(c3c(N)cccn3)=O)C2)ccc(S(N)(=O)=O)s1 24363,N1(C(c2c(C)ncc(Cl)c2)=O)CC2(CCN(C(=O)C3=CCCCC3)CC2)CC1C 24364,N1(C(C(C)OCCC(C)C)=O)CCCN(C(c2cnc3c[nH]nc3c2)=O)C(C)C1 24365,C1(CC)CCOC1C(=O)NC1CC(NC(=O)CC2(O)CCCC2)C1 24366,N1(C(CC(C(C)C)O)=O)CCCCC12CC(NC(=O)COC1CCCOC1)C2 24367,C1(CC(=O)NC2CCN(C(=O)CC3CC4CC4C3)C23CC3)CCS(=O)(=O)CC1 24368,Cn1cc(C(=O)NC2CC3(C2)CC3NC(=O)C=CCC2CCCCC2)ncc1=O 24369,C(=O)(CC(F)(F)F)OC.c12nsc(n1)CCN(C)CCOCCN(C)C2=O 24370,CC(N=c1[nH]c(N(C)CCC2CN(C)C2)nc2c1CCC2)c1nnc2n1CCC2 24371,C(=O)(C1OCCc2ccccc21)NCC1(CNC(c2cnns2)=O)CC12CCC2 24372,C1(CNC(c2cnc(CC(C)C)[nH]2)=O)CCC(CNC(C2CCN(C)C2)=O)CC1 24373,FC1(F)CCC1CNCCCCCc1nc(-c2cccs2)no1 24374,C(=O)(C1CCc2c[nH]nc21)NC(C(NOCC)=O)c1ccccc1 24375,C(C)(CCC(=O)NC1CC1CNC(c1cnc(-c2ccccc2)[nH]1)=O)OC 24376,C1(CNC(C2CC(C)OC2)=O)CC2(CCN(C(C3CC4CCC3CC4)=O)C2)CO1 24377,c1(C(N2C(CC)CN(C(C3(C)CC3)=O)CC2)=O)c(F)ccc(Br)c1Cl 24378,C1(NC(CN(C)CCO)=O)CC2CN(C(=O)C(c3ccccc3)N(C)C)CC2C1 24379,C1(CNC(CCc2cc(C)[nH]n2)=O)(CO)CCN(C(c2sccc2C#N)=O)C1 24380,c1(C(=O)NCC(CC=C)NC(=O)C(F)(F)C(F)F)cc(N)c(O)c(F)c1 24381,C(=O)(C1=NOC(C)C1)N1CCCC(C(C(=O)NCC(=C)Cl)C)C1 24382,C1(C(=O)NC(C)C(C)NC(c2cnoc2-c2ccoc2)=O)CCCC2(CC2)C1 24383,CC1(C)CC(C)(C(N2CC3OCCOC3C2)=O)CN1C(=O)C=Cc1cscn1 24384,C=CC(CC)CC(=O)NCCOCCNC(=O)C=Cc1ccc(C)cc1 24385,n1(C(CC)C)ccc(=NC(=O)CC(CC(C)C)NC(C2C=CCCC2)=O)[nH]1 24386,N1(C(C(C)Cc2ccco2)=O)CCC(OC2(C(=O)NCCN(C)C)CC2)CC1 24387,N1(C(c2c(COC)cc[nH]2)=O)CC2CC(NC(c3ccsc3OC)=O)CC(C2)C1 24388,N1(CCCNC(C(C)OC)=O)CCC(NC(=O)C(C)(F)F)C1 24389,C(=O)(C1CCCc2scnc21)N1CCC(CNC(c2n(C)c3c(c2)scc3)=O)C1 24390,C(C)(CN=c1cc(COC)nc[nH]1)(C(C)C)NC(c1ccc(CC)cc1)=O 24391,C(C)(CSC)(C(=O)NC(c1cccnc1O)C)NC(C1CC(=C)C1)=O 24392,C12CCC(F)(C1)CNC2=O.c1(C2C(N(C(=O)C(C)C)CC)C2)ccc(Br)s1 24393,C(=O)(C(CC)(CC)c1ccccc1)NCC(CCCC)NC(=O)OC(C)(C)C 24394,C1(C(=O)NCCN2CCNCC2)CN(C)CC(C)O1.n1(CC)cc(C2(N)CC2)nn1 24395,C1(C(=O)OC)COC2(CCCCC2)O1.c12ccccc1CNC(=O)COC2=O 24396,Nc1cccc(CC(N2CC(n3cc(-c4cn(CCF)nn4)cn3)C2)=O)c1 24397,C(C(F)(C(=O)NCCC1CCCC(C)C1)C(C)C)NC(COCCC=C)=O 24398,N1(C(C2C(C)(C)C2(F)F)=O)CCC(NC(c2ccnc(N(C)C)c2)=O)C12CCC2 24399,N(C(=NCCF)NCC(N1CCCCCC1)(C)C)CC(N(C)C)C1CC1 24400,C#CCCCCCCCNC(=O)C(CC#C)NC(=O)CNC(=O)CC 24401,C12(CNC(C(C3CCCC3)SC)=O)CC(CO)(C1)C2.C12(CC1)C(=O)N2 24402,C1(C(=O)NC2C(C(NOC(C(C)C)CO)=O)CCC2)COC(=O)N1C 24403,C1(NC(=NCC=C)NCCS(=O)(=O)NC(C)(C)C)CC2(C1)CC(F)(F)C2 24404,N1(C(CCC(C)OCC)=O)CCC(C2CCCN(C(=O)C(=O)C(C)CC)C2)CC1 24405,C12(NC(c3ccc(C)cc3)=O)CC(CNC(=O)CC(O)C(C)C)(C1)OC2(C)C 24406,c1(C(=O)NC2(CO)CN(C(CCc3scc(C)c3)=O)C2)ccc(Br)nc1C 24407,N1(C(c2n(C(C)C)cnc2)=O)CCCCC(N=c2ccc(C(F)(F)F)n[nH]2)C1 24408,C1(NC(c2cnc(CC)[nH]2)=O)(CNC(c2cc3c(s2)CCC3)=O)CC2CCC1C2 24409,c1(C(=O)NCCC2N(C(C(N3CCOCC3)C)=O)CCC2)cc2ccccn2n1 24410,C1(C(=O)NCC(C2CCC2)OCC)CC(O)CN1C(c1ncccc1Cl)=O 24411,C(=O)(C(CO)C(C)(C)C)N1CC(CCNC(=O)Cn2ccc(O)nc2=O)(OC)C1 24412,N1(C(CCCC#C)=O)CCC(C(=O)NCC2(O)CCC(C)C2)C12CCC2 24413,c1(CC(=O)NC(C2CCCN2C(=O)CCC2CC2)C)cn(C2CC2)cn1 24414,c1(SCCNC(=O)NC(=O)CN2CCCC2C(F)(F)F)cc(Cl)ccc1Cl 24415,N1(C(C(COC)OC)=O)CC(CNC(c2cccc(-n3cccc3)c2)=O)CC1C 24416,Cn1cc(C=CC(=O)NCC2(NC(C3CC4C=CC3C4)=O)CCC2)nn1 24417,N1(C(c2cnc(C)c(N)c2)=O)CCC2(CCCC2CNC(C2(Cl)CC2)=O)CC1 24418,c1(C(=O)NCC(C2CC2)NC(c2cc(C(C)C)n(C)n2)=O)cn2c(n1)COCC2 24419,Cc1c(F)ccc(-c2cn(C(C)CNC(c3scnc3C(C)(C)C)=O)nn2)c1Cl 24420,c1(OC(C)C)ccc2ccnc(C(C)NS(=O)(=O)CCCOC(C)(C)C)c2c1 24421,C(N=c1nc2c(ncn2C)c(NC2CC2c2c(Cl)cccc2Cl)[nH]1)c1c(C)occ1 24422,Fc1cc(CCNC(=S)NC(C2CCCCO2)C2CC2)ccc1Cl 24423,N1(C(c2ncc(CC3CC3)s2)C(=O)NCCOCC)CCOC(c2cccs2)C1 24424,C1(CNC(c2ccc(OCC)cc2)=O)CCC(C)CN1C(c1cccc(O)n1)=O 24425,C1(CCNC(c2c(C)ocn2)=O)CCCN(C(C2CCCOCC2)=O)C1 24426,c1(SCC)cccc(C(N2CCC2CNC(=O)C(C(C)C)NS(C)(=O)=O)=O)c1 24427,C1(C(N2CCOCC2CO)=O)CC12CCN(c1nccc(C(F)F)n1)C2 24428,C1(CC)(CC)CC(NC(C2CC2C2CC2)=O)CN1C(=O)CCCF 24429,C(C(=O)NC(C1CCCC1)CNC(=O)CC1CC1(Cl)Cl)(C(C)C)NC(C)=O 24430,c1(C(=O)NC(C)CCCNC(c2cn(C3CC3)cn2)=O)cccc2nc[nH]c12 24431,N1(CC)CC(C(N2CCC2CNC(C2(c3ccsc3)CC2)=O)=O)CC1=O 24432,Cc1ccc(C(N2CCC(NC(=O)CN3CSCCSC3)C2)=O)cc1OC(F)F 24433,N(C(=NCCOc1ccccc1)NC1CC1)C(c1cccc(CS(C)=O)c1)C1CC1 24434,CCC(CC(=O)NC1CC=C(C(=O)NCCCC2CCC2)C1)C(F)F 24435,C1(CNC(CCC=C)=O)(NC(=O)C(O)Cc2cccc(Cl)c2)CCCCC1 24436,c1(C(N2CCC(NC(C(C=C)O)=O)C(O)C2)=O)c(C)cc(O)cc1C 24437,Cc1cc(C(N2CC3(NC(c4nnc(S)n4C)=O)CCC2CC3)=O)cc(N)c1O 24438,C1(C(N2CC(NC(CCSCC(C)C)=O)C3(C2)CC3)=O)CCC2(CC1)CC(O)C2 24439,C(=O)(C1=NNC(=O)CC1)NCC(C)N(C(c1c(C)ccnc1Cl)=O)C 24440,CC1(C)CN(C(=O)C2=CCCCO2)CC1C(=O)NC1CC2C=CC1C2 24441,c1(OC)cccc(C(=O)NCC(C)CNC(c2cnc(CC(C)C)s2)=O)c1N 24442,c1(C(N2CC(C(=O)NC(C3CCCC3)C#C)C(OC)C2)=O)cncc(C=C)c1 24443,C#Cc1ccc(C(=O)NC(C2CCCN2C(c2ccc(=O)n(O)c2)=O)(C)C)nc1 24444,C(=O)(CC(C)C(C)(C)C)NCC1N(C(C(CC(=O)OC(C)(C)C)O)=O)CCC1 24445,c1(NC(C2C(C(N(CC#C)C)=O)C2)=O)cc(Br)cc(F)c1OC 24446,c1(C(=O)NCC2C(CNC(C(C)SCC)=O)C2)c[nH]c2c(C)c(C)ccc2c1=O 24447,Cc1c(C(=O)NCC2(CNC(=O)C(C)CS(C)=O)CCC2)ccc2c1CCC2 24448,c12cccc(c1)CC(=O)N2.C(=O)(C1=CCCC1)N1CC(C)(OCC=C(C)C)C1 24449,c1(SC)nc(OC)cc(OC)n1.C1(N(C(=O)CN2CCCC2)CC)CC2CNC1C2 24450,CC1COCCCN1C(C1CC(O)CN1C(=O)Cn1cnnc1)=O 24451,c1(C(=O)NC2CN(C(C(C)SCC)=O)CC2C2CC2)c(C)[nH]cc([N+](=O)[O-])c1=O 24452,N1(C(C2C(NC(=O)Cc3ccccc3[N+](=O)[O-])C2)=O)CCc2cc(O)ccc2C1 24453,C1(C(N(C)CC2OCCN(C(C3N(C)C(=O)CC3)=O)C2)=O)C(F)(F)C12CCC2 24454,c1(CC(=O)N(CC(CC)NC(C(C)SCC)=O)C)cccc2ncccc12 24455,Cc1n[nH]c(C)c1C(C)CC(=O)NC1CC(C)N(C(=O)Cn2cncn2)C1 24456,C(=O)(N=S1(=O)CCNC(C(F)(F)F)C1)c1ccc(NC(=O)OC(C)(C)C)c(C)c1F 24457,N1(C(C(=O)NCC)=O)CC=C(C(C)(C)C(=O)NCC2OCCC2(C)C)C1 24458,C1(C(c2cn(Cc3nnnn3C)nn2)C)CCN(Cc2cnoc2)CC1 24459,C1(C(=O)OCCC2(CC3CC3)OCCO2)Cc2ccncc2C1 24460,C(CC(C(=O)NCc1ccc(CC)cc1)NC(C1CCS1(=O)=O)=O)=CC 24461,C12(NC(C3OCCC(C)C3)=O)CC(CNc3cc(CC4CC4)ncn3)(C1)OC2C 24462,Cc1ccnc(C(=O)NCc2ncc(C(=O)NCCCn3cccn3)cn2)c1F 24463,c1(OC)cc(CC(N2CCCC2NCCN2CCOCC2)=O)cc(F)c1OC 24464,c1(CNC(=N)NC(c2cccc(Cl)c2)C(F)F)ccccc1Br 24465,c1(C(=O)NC(C2CN(C(N)=O)C2)C)ccc(NC(c2[nH]cnc2C#N)=O)cc1 24466,c1(Cc2ccc(COCC)o2)ncnc2c1ncn2CC(COC)CCCCO 24467,c1(CCCOC)cn(CC(N2CC(SC)C2)=O)nn1 24468,CC1CC(c2nnnn2CSc2ccccc2)(NCC2(CCO)CCC2)CS1 24469,N1(C(C2CC(C)(CC)C2)=O)CC=C(CC(=O)N2CC(F)(F)CC2CO)CC1 24470,N1(C(C(c2ccccc2F)C)=O)CCN(C(=O)CC=C(Cl)Cl)C2(CC2)C1 24471,N1(C(CC2CCC(=O)C2)=O)CC2CCC1CN2C(C1C2C=CSC12)=O 24472,C1(C(=O)NC(CNC(c2nc(C)sc2)=O)(C)Cn2cccn2)CCC(O)CN1C 24473,Cc1nc2ccc(-c3cncnc3C(=O)NCc3nccnc3Cl)cc2[nH]1 24474,N1(CCC(N2CC(F)(C(=O)OCC)C3(C2)CCC3)=O)CCc2ccccc2C1 24475,C1(CNC(C)C(=O)Nc2cccc([N+](=O)[O-])c2)NCCC12CCCCC2 24476,Cc1csc2c(NC3CCC(NC(=O)CC4CCC(C(N)=O)O4)CC3)ncnc12 24477,c1(C(=O)NC2(C(=O)NCc3nc(C)on3)CC2)cc(F)cc(Cl)c1 24478,c1(CN(C)CC2(c3cncc(F)c3)CC2)ccc(-c2nn[nH]n2)cc1 24479,C(=O)(CC(C)(C)C(F)F)N(C1CCN(C(c2cnn(C3CCC3)c2)=O)C1)C 24480,C(CC(CC)C(=O)N1CCCC(N(C)C(C2CCC(N(C)C)CC2)=O)C1)=CC 24481,N=c1[nH]n(CC(=O)NC2CC(NC(C3C4CNC(=O)C34)=O)C(O)C2)cc1Br 24482,c1(C(N2CCC(NC(C3(COC)CC3)=O)C2)=O)c(C)nc2sc(C)cn12 24483,C1(NC(Cn2c(=O)sc(C)c2C)=O)CCCC2CN(C(c3cccnc3)=O)CC12 24484,C1(c2ccccc2)(C(N(CC(O)CNC(C2(CF)COC2)=O)C)=O)CCCO1 24485,c1(C(=O)NCC2(O)CC(NC(c3cncc(C(F)F)c3)=O)C2)cnc2n1CCS2 24486,CC(C)C(C(=O)NCC(C)N(C)C(C1(C)CC1)=O)c1ccncc1 24487,CC1COc2c(C(N3CC(CNC(c4ncccc4N)=O)C3)=O)cnn2C1 24488,Cc1cc(NC(=O)CCN(C(C2CC3CCCC3C2)=O)CC2CC2)cn(C)c1=O 24489,n1(CCC)nc(C)cc1C(=O)N(CC(C)CNC(C1(c2oncc2C)CC1)=O)C 24490,c1(C(=O)NC(C2CCCCN(C(=O)C(F)=CC3CC3)C2)C)cnc(N)c(Cl)c1 24491,Cc1ccc(C(C)NC(c2ccc(Cl)o2)c2nnnn2C(C)(C)C)s1 24492,C1(CC(=O)NC(C(C)NC(CNS(CC)(=O)=O)=O)(C)C)COCCN1C 24493,CN=c1[nH]ccc(C(N2CCC(C)(C)C2CNC(C2CCC(C)CC2)=O)=O)c1N 24494,c1(CNC(C=CCOC)=O)ccc(C(=O)NCCN2CC(CF)C2)s1 24495,CCCCC(CNC(=O)Cn1cc(CO)nn1)NC(C1CCN1C1CCCC1)=O 24496,C#CC1CCCC(NCCCC(N)=O)C1 24497,c1(C(=O)NCCN(C(C2C(C)C2(F)F)=O)C2CC2)cccc(C2(F)COC2)c1 24498,c1(C(=O)NC2(C)CN(C(C3CCN(CC#C)CC3)=O)C2)cnc2nncn2c1C 24499,N1(C(C2CCCC(OC)C2)=O)CC2(CCN(C(=O)C(C)NC=O)C2)C1 24500,N1(C(C(COC)C)=O)CCC2(CC1)CN(c1nnc(C3CC3)s1)CCO2 24501,c1(CC)ccc(C(=O)NCCC2CCN(C(=O)CCCC#N)C2)cc1Br 24502,C1(C(=O)NC2CC(CC)(CC)C2)CN(C(=O)CC(C)SC)CC1N=[N+]=[N-] 24503,c1(NC(c2cn(C3CCCCC3)nn2)=O)ccc2c(O)ncnc2c1 24504,C(=O)(C(C)C(F)(F)C(F)F)NC1(CCCNC(c2cc(CC)c(F)cc2)=O)CC1 24505,Cn1c(C(=O)NCC2CCCC(NC(=O)C=C3CCC3)C2)cc2ccsc12 24506,c1(C(N(C)CC2CCN(C(C(C3CC3)OC)=O)CC2)=O)cc2n(c1)CCC2 24507,n1(CC(=O)NCC(C)(CO)NC(C2CSCC(=O)N2)=O)sc2ccccc2c1=O 24508,CC1CN(C)CC1NC(C1CCN(C(c2ccoc2Cl)=O)C1C)=O 24509,c1(C(N2C(CC=C)C(C)(C)CCC2)=O)ccc2nnn(C(C)(C)C)c2c1 24510,CC1CCNC(=O)C1NC(=O)NCC1CCC(c2ccccc2)O1 24511,C(CC)(CCCC(=O)NCc1ccc(O)cc1)NC(C1(OCC)CCCC1)=O 24512,CCCCC(CO)NC(=O)CC1CC(NC(=O)CN2CCNC(=O)C2)C1(C)C 24513,C1(C(=O)NCCCN(CC)CC)(NC(=O)CCSC)CCOC1 24514,Cc1cc(Cl)c(C(=O)NCC2(C)CCCN2C(=O)CSCc2ccncc2)cn1 24515,c1(N(C)C)cc(NC(C2C=CCN2C(c2cc(C3CC3)on2)=O)=O)ncn1 24516,c1(NCCOC(C)C)[nH]c(=NCC(c2ccccc2)N(C)C)nc2c1ncn2C 24517,CC1CCCC(N=c2nc(N3CC4CCC3CC4)c3c([nH]2)CCOC3)C1 24518,C1(COC)(NC(c2cocc2C)=O)CCN(C(=O)C(C#N)C(C)C)CC1 24519,c1(CC(=O)NC(CC(C)NC(CCOCCC)=O)C)ccc(F)cn1 24520,c1(-n2c(C3C4(CC4)N3)nnn2)csc(CSC)c1OC.C1(SC)CCCCCC1 24521,CCC(C)C(C(=O)NC(C)CCN(C)C(c1cccc(C)c1C)=O)N(C)C 24522,C1(C(N2C(CNC(=O)CN3CSCC3=O)CCCC2)=O)CCC=CCCC1 24523,N1(C(c2cccc(CC)c2)C(=O)NC)Cc2nccn2CC(C(=O)OC)C1 24524,C(=O)(CCC(CF)CF)N1CC(CC(C(=O)NCCC2CC(O)C2)F)C1 24525,C1(NC(c2c(C)scc2)=O)CN(C(C2CCC2C(C)(C)C)=O)C2(CCC2)C1 24526,C(CS(=O)(=O)CC(=O)NC(C)(C)CC(F)C(=O)NCc1nnnn1C)OC 24527,C1(C(=O)NC2COCC2F)(COC)CCCNCC1 24528,c1(CC(=O)NC)ccc(OC)cc1Cl.C12(C(=O)OC(C)C)CCC1CN2 24529,Cc1c[nH]c(C#N)nc1=NCC1CCCN(C(=O)C2=CC3(CCOC3)C2)CC1 24530,Cc1ncc2n1CCC(C(=O)NCCNC(=O)CCc1ccc(CO)cc1)C2 24531,C1(NC(C(CCCCC)O)=O)CCN(C(c2cccnc2OC)=O)CC12CCC2 24532,c1(C(C(=O)NC(C)CN(C(=O)CSC(=N)N)C)C)cccc(O)c1 24533,CON1CCC(CC(=O)NC2CCC(NC(c3c[nH]c(C#N)c3C)=O)CC2)CC1 24534,Cc1cccc(C(O)C(=O)NCC2(CNC(C3(N(C)C)CC3)=O)CCCC2)c1F 24535,N1(C(C(CCF)NC(C2CCC(=O)OCC2)=O)=O)CCC2(CCC2)CC1 24536,c1(CCCC(=O)NC(CNC(C2CCOC2)=O)C2CCC2)ccccc1Cl 24537,C(=O)(C(F)(F)C(O)C1CC1)NCC12N(C(C(C=C)O)=O)CC(C1)C2 24538,C(=O)(CC(C)(C)c1ccccc1)NCC(CCOC)NC(=O)C(F)=CCCF 24539,C1(CC)CC(N=c2[nH]c(=NCc3nncn3C3CC3)c3cccc(F)c3[nH]2)C1 24540,N1(C(CC(C(C)C)NC(CC(=O)OCC)=O)=O)CCn2ccnc2C1C 24541,c1(C(=O)NCC(C2CCC2)NC(CC2C(C)(C)C2)=O)cocc1Br 24542,N1(C(c2ccc(C)cc2)=O)CCC(NC(C2CCC(CO)CC2)=O)C(F)C1 24543,C=CC1(CC(=O)NCC(C2CCN(C(C3CCC(=O)O3)=O)CC2)F)CCCCC1 24544,n1(CC=C)nc(-c2cccc(Br)c2)nc1C1CCCC1O 24545,C(=O)(C(F)C(C)CNC(c1ccc(F)c(O)c1)=O)N1C(COC)C=CC1 24546,C(=O)(C(C)(C)C(=O)Nc1cc(F)cc(F)c1)NCC1(O)CCN(C(C=CC)=O)C1 24547,Cc1ccc(F)cc1C(N1CCC(N(C(=O)CC2(O)CCCCCC2)C)C1)=O 24548,C(=O)(C(F)C(F)(F)F)N(CC(O)CNC(=O)Cc1cccc(C(F)F)c1)C 24549,Cc1c(Br)cnn1CC(=O)N(CC(C)NC(=O)C(F)=C1CCC1)C 24550,CC(C)CS(=O)(=O)CCC(=O)NCC(C)CN(C(=O)CP(C)(C)=O)C 24551,CC1(C)CC(CC(N2CC(CC(F)F)C2)=O)N(CCNC(=O)CO)C1 24552,C1(C(=O)NCC(C2CCC2)OCC)CC(F)(F)CN1C(=O)CCc1cn[nH]c1 24553,CCCCCC(CC)C(=O)NC1C2CCC1N(C(=O)C=Cc1cccc(Cl)c1)C2 24554,c1(N2C(C)CC(NC(c3cc(Cl)on3)=O)CC2)ncc([N+](=O)[O-])cn1 24555,N1(C(=O)CSCCNC(C2C=CCS2)=O)CC=CC12CCCCC2 24556,N1(C(c2cc(F)cc(C)c2N)=O)CCOC2(C1)CN(C(C1CN(C)C(=O)N1)=O)C2 24557,Cc1cc(CCC(N2CCCC(N(C(=O)C(C3CC3)C3CC3)CCO)C2)=O)nn1C 24558,N1(C(C)C)CCCC(NC(c2coc(CNC(=O)Cn3cccn3)c2)=O)C1 24559,N1(CCn2cc(CNC(=O)OC)nn2)Cc2ccc(F)cc2CC1C 24560,C1(C(=O)NCCN(C(C(CC=C)C(C)C)=O)C)CCOC2(CCOCC2)C1 24561,c1(C(=O)NC2CC(CNC(Cc3nnc(C)n3C)=O)CC2O)c(C)ncnc1O 24562,c1(-c2c(C(=O)Nc3ccc(F)cc3O)n[nH]c2)ccc(S(=O)(=O)N2CCCC2)cc1 24563,C1(NS(CC=C)(=O)=O)CC2(C1)CN(C(c1cc(I)ccc1O)=O)C2 24564,C1(CC(=O)NCCCC(C)NC(Cc2cccc(OC)c2)=O)CCCC(C#N)C1 24565,CC1(C)CN(C(=O)CCn2ccnc2)CC(C)(C)C1NC(c1ccc[nH]1)=O 24566,C1(NC(=O)CN2CCOCC2)CCN(C(=O)CCc2cn[nH]c2)CC1F 24567,C(=O)(CC(O)CC(C)C)N1C(CCC)CN(C(=O)CC(C)F)CC1 24568,C(C1CCN(C(C2CCCN2C=O)=O)CC1)=CC(=O)NC(C#C)(C)C1CCOC1 24569,C1(c2c(C)cco2)NC(=S)N(Cc2ccco2)C2=C1C(=O)NC2(C)C 24570,C(C(=O)N1OC2CCC1CC2)N(C(=O)C(F)C1CCCC1)CCOC 24571,C1(N2C(c3nc(C)nc(=N)[nH]3)CCC2)CCC2(CC1)OCCO2 24572,C(C)(CCCNC(=O)C(C)Sc1nncn1C)NC(C1(CCC=C)CC1)=O 24573,c1(NCc2c(OCC)cccc2)ccc(Nc2ncc(C(=O)OC)cn2)cc1F 24574,Cc1ccc(C(F)(F)C(N2CC(NC(c3cnc(C)o3)=O)C(C)C2)=O)cc1 24575,C1(O)(CCNC(C=C(COC)C)=O)CCN(C(=O)Cc2cnc(C(C)C)[nH]2)C1 24576,C=C=C(C)CC(=O)N1CCC(O)(C(C)NC(=O)Cc2c(C)n[nH]c2C)C1 24577,CCCC(C)CC(=O)N1CC(NC(=O)CCCc2ccccc2)C(O)C1 24578,N1(C(C2SCCN(C(CN(C)C)=O)C2)=O)CCN2C(=O)CCC2C1 24579,c1(C(N(CC(N2CC=C(COC)CC2)=O)CC)=O)ccc(=O)oc1 24580,N1(Cc2nccc(C(=O)OC)c2)CCC(NC(=O)Cn2cc(Cl)cn2)C(C)(C)C1 24581,C(=O)(C(O)C(C)CC)NCC1(C(C)NC(CNS(CCCC)(=O)=O)=O)CC1 24582,N1(C(C(CC)NC(N)=O)=O)CC2CC2C1C(=O)NCc1nccn1C(C)C 24583,c1(NC(CC(C)F)=O)sc2c(c1C(=O)Nc1ccccc1)CCCC2 24584,c1(OC2(C(=O)NCC(c3cccc(F)c3)C)CC2)ccc(Cl)cc1 24585,N1(C(=O)CCC2CCCN2Cc2cncc(Cl)c2)CCc2c(Cl)ccc(Br)c2C1 24586,N#Cc1c(N2CCC(F)(CNC(C34CC=CCN3CCC4)=O)CC2)cccc1F 24587,c1(C(N2CCC(O)(CCNC(C(C)C)=O)C2)=O)nc(N(C)C)nc(=N)[nH]1 24588,Fc1cc(Cl)cnc1-c1nnc(N2CC3CN(CC(F)(F)F)C3C2)o1 24589,C(=O)(C(C)(CNC(=O)CCc1nc(O)n[nH]1)CC)NCC(N(OCC)C)=O 24590,C(=O)(C(C)C(C)CC)N(CC(CNC(c1nc(C(=O)NCC=C)sc1)=O)(C)C)C 24591,c1(C(=O)NCC2OCCCN(C(COCCC#C)=O)C2)cccc2nc(O)[nH]c12 24592,N1(C(CC(=O)NC)=O)CCC2(CC1)CCN(C(c1ccc(CC(C)C)cc1)=O)C2 24593,c1(C(=O)NC23CCN(C(=O)Cc4nc[nH]n4)CC2C3)ccc2ccsc2c1 24594,N1(C(CCCSC)=O)CC2CCCC(NC(C3CCCC34CC4)=O)C2C1 24595,CC#CCCCC(=O)NCCOCCCNC(=O)C(c1ccn(C)n1)C 24596,C(=O)(C(CCC(C)C)NC(c1ccnn1CCC)=O)NC(C=C)C1CCC1 24597,CCC(O)C(C)C(=O)N1CCC2(CC2NC(=O)CCc2cn(C)cn2)C1 24598,c1(OC)ccc2nc(N3CC(CO)(NC(c4c[nH]nc4C)=O)C3)sc2c1 24599,N1(C(c2c(SC)cn(C)n2)=O)CC(C)(CNC(=O)C(F)(F)C2CC2)CC1(C)C 24600,N1(C(C2=CC(C)(C)C2)=O)CC2(C1)CN(C(c1cccc(CCO)c1)=O)CC2CO 24601,CCC(C)(CO)C(=O)NCCC1CC(NC(=O)C(C(C)C)n2cnc(C)c2)C1 24602,C1(C(N2CCC(CNC(c3ccc(CO)o3)=O)C2)=O)CCC=CCCC1 24603,c1(OC)cccnc1C(=O)N(C(CNC(=O)CCSc1nnnn1C)C1CC1)C 24604,N1(C(c2ccc(C)nn2)=O)C2CCC1C(CNC(c1cnc(C3CC3)s1)=O)C2 24605,C(C(C)(O)CC)NC(C1(CCNC(CC2CC(=C)C2)=O)CCC1)=O 24606,CC1CCCC1CC(=O)N(CCCN(C(=O)CCCc1n[nH]c(=N)s1)C)C 24607,C(=O)(C(C)(C)C(C)(C)C)NCC1(C(=O)NCc2cccc(C)c2O)CC1 24608,Cc1ncnc(C)c1CC(N1CCC(F)C(NC(C2CCC3CC2CO3)=O)C1)=O 24609,C1(C(=O)NC(CN(C)C)CCO)(CC)CCN(C(c2ccon2)=O)C1 24610,N1(C(C2C(C)CCN2C(=O)CCC(N)=O)=O)CC2(CCCCCC2)C1 24611,c1(C(N(c2cc3ncnn3cn2)C23CC(N)(C2)C3)=O)[nH]nc2ncccc12 24612,c1(-c2c(C)ccs2)ccc2c(c1NC(=O)Cn1cccn1)OCO2 24613,C1(NC(C(CC2CC2)OC)=O)CC2CC(C1)CN(C(=O)Cc1ccc(O)cc1)C2 24614,N1(C(C2CC(n3cc(C4(CO)CCCCC4)nn3)C2)=O)CC2CCCC(C2)C1 24615,CCC(F)(F)C(=O)N1CCOC(CCNC(c2cnnn2C2CCOCC2)=O)C1 24616,N1(C(C(C)CCO)=O)CCOC2(CCCN(C(c3cc(Cl)ncc3F)=O)C2)C1 24617,c1(OCC(=O)NCCC2CC(NC(=O)CC3(C)CC3(F)Cl)C2)cccnc1 24618,N12CCC(OC)(C1)C2=O.C1(=O)C(C(=O)C(C)=O)NCCN1C.C(C)(C)(C)N.OCC 24619,Cc1ccccc1C(C)C(N1CCC(N(c2nncs2)CCO)CC1)=O 24620,C(=O)(C1=NNC(C(F)(F)F)C1)N(CCCNC(C(C)SCCCC)=O)CCO 24621,N1(C(C=CCC)=O)CC(CNC(C23CCC(C)(CO2)C3)=O)CC12CCOCC2 24622,CCC(CN(C)C)C(=O)NC(C)CCCNC(=O)C(C)(C)N(C)C 24623,C1(C(N2CC(OC)(CNC(=O)C(C)(C)c3ccccn3)C2)=O)CC1C1CCCC1 24624,C(CCC(=O)N1CC2(CCC2O)C1)(C(C)C)NC(c1cccc(CC)n1)=O 24625,c1(C(=O)NCC(CC)(CC)NC(=O)C(O)C(C)SC)nc2n(c1Cl)CCCC2 24626,N1(CC(N2CCC(CNC(C(c3ccccn3)C)=O)C2)=O)CCC(=O)CC1 24627,CC1CC(CC(N2CCC(C3(C)N=N3)C2)=O)CN1C(=O)CSCCN(C)C 24628,c1(C(N2CCC(N(C(=O)CC3CCOC3)CCC)C2)=O)cccc2c1OCCO2 24629,c1(CN(C(=O)Cc2ccnn2C2CCOCC2)C)cccc2c1OC(F)(F)O2 24630,N1(C(CN(c2ncccn2)C)=O)CC2CC2(C(=O)NC2CSC2)C1 24631,N1(C(CSC(=N)N)=O)CCn2ncc(C(=O)NCc3ccc4nncn4c3)c2C1 24632,C1(C(=O)NCC(CO)NC(c2n(C)cc(C(F)(F)F)c2)=O)CC2CCCC(C1)C2 24633,c1(C(C(=O)NCC(C)NC(C2CC2[N+](=O)[O-])=O)C)cncc(F)c1 24634,Cc1cc(C(=O)NC(c2ccccc2)C(C)NC(=O)CCC2CC2)nc(O)n1 24635,N1(CC(=O)N(S(CC2CCC(C)O2)(=O)=O)C(=O)C2CC2)CC2(CCCC2)C1 24636,N1(C(C(CC)OC)=O)CCCC(F)(C(=O)Nc2cn(C)nc2C#N)C1 24637,C1(C(=O)N(CC)Cc2ccc(C)o2)(OCC)CCN(C(C)C)CC1 24638,N1(C(C(C)c2ccco2)=O)CCCN(C(c2ccc(Br)s2)=O)CC1CO 24639,C1(NC(=O)C=Cc2cnc[nH]2)CC2CC(NC(=O)CCc3cc[nH]n3)CC2C1 24640,Cc1cc(C(=O)NCCC2(C)CCN(C(c3nnn(C)c3N)=O)CC2)ncc1Cl 24641,C(C1CCN(C(C2CCCC(=O)N2C)=O)CC1)=CC(=O)NCc1c(CC)nccn1 24642,C1(NC(C(Cc2ccoc2)NC(CCCCN(C)C)=O)=O)CCC(N=[N+]=[N-])CC1 24643,Cc1nn(C)c(C(=O)NC(C)CCNC(=O)C(C(C)C)N2CCN(C)CC2)c1Cl 24644,C(=O)(C(CCF)NC(=O)CCOC1CC(OC)C1)NC(CCC)CO 24645,C1(CC(=O)NCCC2CCN(C(C3(O)CC(F)(F)C3)=O)C2)CCCOCC1 24646,c1(C(=O)NCC2CCC(NC(c3cc(C)on3)=O)C2)cc2c(C)cc(F)cc2[nH]1 24647,N1(CC)CCOC(C(N2CCOC(CNC(=O)CC(F)(F)Br)C2)=O)C1 24648,CCN=C(NCC(CO)C(C)(C)C)N1CCC(COc2cccc(C)n2)CC1 24649,C(=O)(CC(C(F)F)NC(c1c(O)noc1C)=O)Nc1ccc(OC)nc1 24650,Cc1oc(C(=O)NCC(O)CN(C(=O)Cc2cnnn2C)C)cc1CO 24651,Cc1ccc(F)c(C(=O)NNC(=O)N(c2cccc3[nH]ncc23)C(C)C)c1F 24652,N1(C(C2CC(N(C)C)C2)=O)CCC(NC(C2CCC(F)(F)CC2)=O)C(O)C1 24653,N1(C(CN(CCC)C)=O)CC(C(=O)NCc2ccnc(Cl)c2)C2(CCC2)C1 24654,C1(C(=O)NC2CC(CNC(c3c(OC)nccc3)=O)CC2O)CCCC(=O)N1C 24655,C(C)(C)(CCC(=O)N(C)Cc1ccon1)NC(C(CC)NC(N)=O)=O 24656,Cc1nccc(C(=O)NCCOC2CCN(C(C3CCC(C)NC3=O)=O)C2)c1C 24657,c1(C(=O)NCC2C(C)CN(C(c3cccc(C(N)=O)c3)=O)C2)c(F)ccnc1F 24658,N1(C(C(CC)NC(=O)CCc2cccn2C)=O)CCOC(C)CC1 24659,C1(CNC(CSCC)=O)CCC(C)CN1C(c1ccnn1CC(C)C)=O 24660,C1(C(C)(C)NC(=O)C=C2CC2)CCCN(C(c2ccc(C(N)=O)cn2)=O)C1 24661,C1(NC(=O)C(O)C2CCCC2)CC2CN(C(c3occc3C3CC3)=O)CC2C1 24662,C(C)(C(=O)NC1(C(=O)NCCC(C)N(C)C)CCC1)OCCC#C 24663,c1(NC(CN(C(=O)C(C)C2CCC2)CC)=O)cscc1C 24664,C(C1CC(=O)Nc2ccccc21)NC(=NCC)NC1CCS(=O)(=O)C1 24665,Cc1ccc(C(=O)NC2CCN(C(=O)CC3(C)OCCO3)C2)cc1[N+](=O)[O-] 24666,C12(C(N(CC(CN(C(=O)C(=O)Cc3ccccc3)C)O)C)=O)CCOC(C)(C1)C2 24667,Cc1c(NCCCN(C)CCOCCC(C)C)ncnc1Nc1ccc(F)cc1 24668,N1(C(CC=C=C)=O)Cc2ccnn2CC(NC(=O)C(C)CCOC)C1 24669,C(=O)(C(C)(C(F)(F)F)c1ccccc1)NCC(=O)NCC(C1CCCCC1)CO 24670,N1(C(CC=CC(C)(C)C)=O)Cc2ccccc2C(NC(=O)CC2CCC2(F)F)C1 24671,CC(C)C(C)(C)C(=O)NCC(CC1CCCC1)C(=O)N(C1CCCN(C)C1)C 24672,c1(C(=O)NC2(c3cn(C(CC=C)CC=C)nn3)CCC2)ccc2occc2c1 24673,c1(N2CC(CC(C)C)OCC2)nc(=NCC2CCC2)[nH]c2ccc(Cl)cc12 24674,N1(C(C(C(C)C)NC(=O)OC)=O)CCCC(O)(CNC(C2SCCS2)=O)CC1 24675,C1(CC2(OC(=O)C3CC3)CCC2)CCCN(C(=O)CN2CCCC2=O)C1 24676,Cc1occc1C(=O)NC1CC(C(F)F)(NC(C2CSC2)=O)C1 24677,CC1(C)CN(Cc2cn(Cc3ccccc3Cl)nn2)C1c1cccnc1 24678,C1(CCN(C(CC(C)F)=O)C)CCN(C(=O)CC2CCC23CCC3)CC1 24679,c1(C(=O)Nc2nnc(Sc3cnc(C)c(Br)c3Cl)s2)ccc(O)c([N+](=O)[O-])c1 24680,c1(C(=O)NCCC(C)NC(c2cc[nH]n2)=O)cc2c(s1)CCCNC2=O 24681,c1(C(=O)NCC(NOCC)=O)ccnc(CNC(=O)C(C)(O)CC)c1 24682,c1(NC(C)C)ccc(C(=O)N(C)CC2CCCN2C(c2ncc(Cl)n2C)=O)cc1 24683,c1(C(=O)NCC2C(NC(=O)Cc3ccc(F)c(F)c3)CC2)cc2c(s1)CCCC2 24684,C1(F)(c2cn(CCC(C)C)nn2)CCN(C(C2CC3(CC3)CO2)=O)C1 24685,C1(CC)C(NC(=O)CC(C)OC(C)C)CCCN1C(=O)COCCOC 24686,N(C(=NCCC(C)=O)NCc1ccc(Cl)cc1F)C1CCC(C#C)CC1 24687,Cc1cn2c(n1)CC(C(=O)NCC1CC13CCN(C(c1nncs1)=O)CC3)C2 24688,C(=O)(CCCC(F)(F)F)NCC1CN(C(C2C(C)(C)C(F)(F)C2)=O)CC12CC2 24689,c1(C(COC(C2(CCC=C)CC2)=O)=O)nnn(C)c1N 24690,N1(C(c2nc(C(C)N)sc2)=O)CCOCC1CNC(c1cnn(C)n1)=O 24691,C1(C(N2CCCCC2CN(C(=O)C(C)NC(C)=O)C2CC2)=O)(COC)CCCCC1 24692,N1(C(C=CC)=O)CC2CC1CN2C(=O)CC1NC(=O)CNC1=O 24693,c1(C(=O)NC2CCCN(C(C3C(C)C3)=O)C2)ccc2c(c1)CC2 24694,c1(C(=O)NCc2nc(CNC(C3(C)C=CCCC3)=O)sc2)ccc2c(c1)CC2 24695,C1(NC(c2ccc(NC(C)=O)cc2)=O)CC2(C1)CN(C(c1ncn(C)n1)=O)C2 24696,C1(CC(C(=O)ON2CCCCC2)NC(N(C)CC)=O)CCC(C)(C)CC1.C(C)(C)(C)O 24697,N1(C(CC(COC)C)=O)CCCC2CN(C(c3ncc(C)cc3C)=O)CCC12 24698,N1(C(c2cc(C(=O)OC)oc2C)=O)CCCC2(CCN(C(=O)C(F)C(C)C)C2)C1 24699,c1(CC)cccc(C(=O)NC(C2CCN(C(=O)CS(=O)(=O)N(C)C)C2)C)c1O 24700,N1(C(Cc2c(C)cco2)=O)CCCC12CCN(C(C1(CC(F)(F)F)CC1)=O)C2 24701,c1(CC(=O)NC2CC(NC(c3cnn(-c4ccccn4)c3)=O)C2)ncncc1Cl 24702,N1(CC(C)O)CCC(NC(=O)CCCc2ccc(Cl)cc2)C(C)C1 24703,C1(C(N2CC(OCC)(CNC(=O)CCS(C)=O)C2)=O)CCCCC1(F)F 24704,c1(-c2cn(C3CC(NC(=O)Cn4cccnc4=O)C3)nn2)cccc(Cl)c1Cl 24705,C#CCCC(O)C(=O)NCCC1CCN(C(c2ccsc2)=O)C1 24706,c1(C(=O)NCC2CCN(C(C3C(=C)CC3)=O)C2)cc2sccc2s1 24707,N1(C(CC(C)(F)F)=O)CC2CC(NC(c3ccnc(C(F)F)c3)=O)CC1C2 24708,C1(NC(C(C)=C2CC2)=O)CC2(C1)CN(C(C1(C(C)C)CC1)=O)C2 24709,CC(C)CC(C)C(=O)NCCN1CCN(C(c2csnn2)C)CC1 24710,C1(C)(C(N(CC(CC)NC(c2ccc(CN(C)CC)o2)=O)CC)=O)CCNC1=O 24711,N1(C(C2C(CC)CCO2)=O)CCN(C(c2c(C)cc(C)nc2S)=O)CC(O)C1 24712,N1(CCOc2ccc(OC)cc2)C=NC2=NC(C(c3ncsc3Br)C)C(=O)N12 24713,CCC(CC(=O)NCCN(C(C1CCC=CCC1)=O)C1CC1)C1CC1 24714,N1(C(CCSC)=O)CC(CNC(c2cc(I)c[nH]2)=O)C2CC12 24715,N1(C(C(C2CC2)SC)=O)CC(NC(c2ccc(F)c(Br)c2)=O)CC(F)C1 24716,C(=O)(C1=CCS(=O)(=O)C1)N1CCC(OCC(=O)NCCOC2CCOC2)C1 24717,Cc1c(C(=O)NCCC2(O)CN(C(=O)C(c3ccccn3)C)C2)cccc1N 24718,N1(Cc2cc(C)nn2C)CCC2(CC1)CN(C(C1CC(C)CO1)=O)CCO2 24719,C1(CCC(C(=O)NCC)N2CCC(C(C)OC)CC2)CCC(F)(F)CC1 24720,CCC(CC(=O)NC(C(N1CCC(OC(C)C)CC1)=O)c1ccco1)SC 24721,n1(C(C)(C)C)ncc(C(=O)NC2(CNC(=O)CC3C=CCC3)CCC2)c1N 24722,C1(CC(=O)NCCC(C)N(C(C(CCSC)O)=O)C)CCCCCCC1 24723,c1(C(=O)NCC)ccc(C(N2CC(OCCNC(c3cnc(Cl)s3)=O)C2)=O)s1 24724,c1(N(CCN(C(CC2(CC)CC2)=O)C)C2CC2)cc(C(F)(F)F)nc(Cl)n1 24725,N1(C(C(C)NC(N)=O)=O)CCN(C(=O)Cc2csnn2)CC12CC2 24726,c1(CC)nccnc1C(=O)NC(C)CCNC(c1ccccn1)=O 24727,C(=O)(CC(CC=C)NC(=O)C(C1(O)CCCC1)F)NC1(CC=C)CC=CC1 24728,c1(C(=O)NCCCCC2(NC(C(C)n3ccnn3)=O)CC2)cc2cccnc2[nH]1 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24765,N1(c2n(CCC#C)c(C3CCc4c[nH]nc4C3)nn2)CCCC2(CCCC2)C1 24766,c1(NC)cnncc1C(N1CCC(O)(CN(C)C(C2CC=CCC2C)=O)C1)=O 24767,c1(CC)nc(CCN2CCOCC2)nn1-c1ccn(C)n1 24768,N1(C(C2CN(C)C2)=O)CCC12CCCN(C(c1ccnc(OC(C)(C)C)c1)=O)C2 24769,N1(C(CC=CCC)=O)C2CCC1CC(N(C(=O)COC(C)(C)C)C)C2 24770,N1(C(c2n[nH]c(CC)c2[N+](=O)[O-])=O)CC(C2CCCN(C(=O)C#CC3CC3)C2)C1 24771,N1(C(C(C)OCCC=C)=O)CCCCCC1C(=O)NCC1(OC)CC1 24772,c1(C(N2C(CNC(=O)NC)CCC2)=O)cc(Br)ccc1O 24773,CCC(CO)C(=O)NCCCCCn1cc(COCCOC)nn1 24774,C(=O)(CCCCC(=O)NCC1(C(C)NC(c2cnc(N)cn2)=O)CC1)NC 24775,Cn1cc(N)c(C(=O)N(C2CCN(C(c3ccc(Cl)s3)=O)C2)CCO)n1 24776,S(=O)(=O)(c1ccnc(NC(c2cncc(CN)c2)=O)c1)NC 24777,c1(C(N2CC(O)(CCNC(C(C=C=C)C)=O)C2)=O)cc(Br)c2ncccc2c1 24778,c1(CN(CCOCCOC)Cc2cscc2C)ccccc1 24779,C1(CC(=O)NC(C2CCCC2)CNC(CCc2n(C)cnc2)=O)CCC=CCC1 24780,Cc1ccc(F)c(OCC(=O)N(CC(C)NC(c2ncn3c2CCC3)=O)C)c1 24781,C1(C#N)(C(=O)NC(C(C)C)CNC(=O)CC2CC2C)CC2CC2C1 24782,n1(C(=O)OCC(=O)NC)cc(CN2CCCC2)nn1.C12CN(C1)N2CC.C(C)=O 24783,Cc1cc(Br)cc(C(N2CCC(C)(C)C(NC(C34CC(F)(C3)C4)=O)C2)=O)c1N 24784,c1(C(=O)NC2C(C)CCN(C(c3cnc(C)o3)=O)C2)cc2c([nH]1)CCCC2 24785,N1(C(c2c(CC)occ2)=O)CCC2CCN(C(c3cn(C(F)F)cn3)=O)CC2C1 24786,c1(N2CC(NC(c3cccc(C#C)c3)=O)C(C#N)C2)ncnc2sc(Br)cc12 24787,Cc1c(C(=O)NCCCOCCNC(=O)CC(C)c2ccco2)ccn1C(C)C 24788,CCCC(C(=O)N1CC(NC(C2COCCOC2)=O)CC1CO)OC 24789,c1(OC)cc(C(=O)NC(C)CN(C(=O)C(C)CC2CCC2)C)ccc1SC 24790,CC1(C)COc2cc(CNC(N3CCCC3c3nnc(O)o3)=O)ccc21 24791,c1(-c2nc(N(C(C)=O)C(c3nccnc3Br)=O)sc2)cn(C)nc1C(F)(F)F 24792,N1(C(c2c(OC)n[nH]c2)=O)CC(C)(CNC(C2CC3CCC2CC3)=O)CC1(C)C 24793,C1(C(=O)NCCC(C)N(C(C(C)Cc2ccncc2)=O)C)C2CC3C(C2=O)C13 24794,N1(C(C(CCNC(=O)CCC(F)(F)F)OC)=O)CC(C)(C)CCC1C 24795,C1(C(=O)NC23CC(CCC)(C2)C3)CC(=O)CN1C(=O)C(CC)N(CC)CC 24796,Cc1ncc(N)cc1C(=O)N(C1CCCN(C(C2CC3CCC2CC3)=O)CC1)C 24797,CN1CCN(C(=O)C(C)(C)CC2CC2)CC1CNC(=O)C(F)(F)c1cccnc1 24798,c1(C(N(C(C)CNC(=O)CSC(C)C)CC)=O)cccc(CCO)c1 24799,C1(NC(c2c(CC)cncc2)=O)COC2(CCN(C(c3cn(C)c(C)n3)=O)C2)C1 24800,C1(C(=O)NC(CC=C)CO)CN(C(c2ccns2)=O)CC1C(C)C 24801,C1(C(N(CCCN(C(=O)C=C2CCCC2)C)C)=O)CCC2COCCC2C1 24802,c1(C(=O)NC2C(C)CCN(C(c3ccc(=N)[nH]n3)=O)C2)cnc2ccnn2c1 24803,C(=O)(C1=NOC(CNC(C2CC3COCC3C2)=O)C1)N1CCC(O)(CC(C)C)C1 24804,N1(C(C2(CC)COC2)=O)CC(C)CC1C(=O)Nc1cccc(F)n1 24805,C1(C(=O)NC(CNC(c2n(C)cnn2)=O)C(C)(C)C)CCCCN1N=O 24806,N1(C(C(C2CN(C(c3cc(C)sn3)=O)C2)O)=O)CC(O)CC(O)C1 24807,c1(OC)cc(Cl)ccc1NC(=O)C(C)CNC(=O)CN1CCCC1C 24808,N1(C(C(C)(C)C2CC2)=O)CCOCC(NC(C2(CSC3CC3)CCC2)=O)C1 24809,N1(CC(=O)Nc2c(CN)cccc2)CCOCC(S(N)(=O)=O)C1 24810,C=CCCCC(C(=O)N=c1cc2n([nH]1)CCCC2)NC(c1nn(CC)nc1C)=O 24811,Cc1cc(CC(=O)NC(C)CCNC(=O)CC2CCOC(C(C)C)C2)c(C)o1 24812,c1(C(C(=O)NCc2ccccc2)N(c2nnn(C)n2)C)c(Cl)nc2sccn12 24813,N1(C(C2=CCC(NC(C(CCC)=CCC)=O)C2)=O)CC2CCCCC12C 24814,C1(C(=O)NC(C2CCCC2)CNC(C2NC(=O)OC2)=O)CCS(=O)CC1 24815,CC1(C)CC2(CN1Cc1cccc(OCC(F)F)c1)CC(F)(F)C2 24816,c1(Cn2cc(C3(C)CN(C(c4cnc(C)s4)=O)C3)nn2)cccc2ccccc12 24817,N1(C(c2n(CCCC)ncc2)=O)CC(NC(c2cc(O)ncn2)=O)CC(O)C1 24818,N1(C(C2CCN(C(C(CC)COC)=O)C2C)=O)CCC(O)C(O)C1 24819,CC1CCc2n[nH]cc2C1C(=O)NC1CC2CCC(C1)N2CCS(C)(=O)=O 24820,CCCC(CCC)CCCC(=O)N(CCCNC(=O)CC(C)(CC)C(=O)OC)CC 24821,n1(CC(=O)NC2C(NC(C(C)C(F)(F)F)=O)CCCC2)ccc(=O)n(C)c1=O 24822,N1(C(C(C)CC(C)(C)C)=O)CCC2(CC1)CCN(C(C1COC(=O)N1)=O)CC2 24823,c1(C(N2CCC(CN(C(Cc3ccc(C)s3)=O)C)CC2)=O)cc2c(ncn2C)s1 24824,N1(C(c2csc(-c3ccccn3)n2)=O)CCC2C(CCCN2C(=O)C2CC2)C1 24825,N1(C(CNC(CNC(C(CCC)N(C)C)=O)=O)=O)CC(OC)CC(C)C1 24826,CC1CCN(C(=O)CSCC(F)(F)F)CC1NC(C1(CCF)CC1)=O 24827,C1(c2cc(C)no2)CCCCCN1C(=O)CC1CCN(C(=O)OC(C)(C)C)C1 24828,CCC(CC)C(C)C(=O)NC1CCC(C)(CNc2nc(C(=O)OC)ns2)CC1 24829,c1(CNC(CC2(C)CCN(C(=O)C(F)(F)C3CC3)C2)=O)cnc(O)c(F)c1 24830,C1(CCOC)CCCN(C(c2ccc(NCC(N)=O)cc2)=O)C1.C1(C)CC(=O)N1 24831,N1(C(C(N(C)C)C2CC2)=O)CCC2C(C1)NC(=O)CN2C(=O)Cc1cncn1C 24832,c1(-c2c(C)ccnc2)cccc2c(C(=O)NCCCO)n[nH]c12 24833,C1(C(=O)NC(C(C)NC(c2ccn(C3CCCC3)n2)=O)CO)CCOC(C)(C)C1 24834,c1(C(=O)NCC2N(C(CNC(C)=O)=O)CCCC2)ncc(Cl)cc1Br 24835,C1(C(=O)NCC(CO)NC(c2ccc(C(=O)OC)cc2)=O)CC(C)(C)CN1C 24836,C1(CC(N2CCC(OCC)CC2)=O)CN(C(=O)CN2CCOCC2=O)CCC1C 24837,N1(C(c2ccc(C#C)cc2OC)=O)CCCC12CCCN(C(C1CCOC1)=O)C2 24838,O=C(CCCC(F)F)NCCC12CCC1CN(C(=O)Cn1cc(Cl)cn1)C2 24839,C1(CNC(=O)C(O)C2CC2)CCC2(CCN(C(C3(CCO)CC3)=O)CC2)O1 24840,N1(C(CCOCC#C)=O)CC=CC1CNC(=O)C(C)OCCN(C)C 24841,Cc1ccn2ncc(C(=O)NCC3(F)CCN(C(=O)C(C)OCC4CC4)C3)c2n1 24842,N1(C(=O)Cc2cccnc2O)CCN(C(=O)COc2ccccc2)C(C2CC2)C1 24843,C12(C(=O)NC(CC)CNC(c3cnc(NC4CC4)s3)=O)CCC(CC1)C2(C)C 24844,Cc1c[nH]cc(Br)c1=NC(=O)C1CCCC(NCc2nccn2C)C1 24845,c1(C(=O)NC2(CNC(C(C)OC3CCCCCC3)=O)CC2)ccc(P(C)(C)=O)o1 24846,c1(C(=O)OC)ccc(C(=O)NCC(C)NC(=O)CCC(C)SC)cc1Cl 24847,c1(C(=O)NCC(CC)NC(=O)Cc2cc(F)ccc2Cl)cc(F)c2cn[nH]c2c1 24848,c1(C(N(CCN(C(=O)CC2C=CS(=O)(=O)C2)C)C)=O)cccc2[nH]ccc12 24849,C1(NC(C2(CC(=O)OC)CC2)=O)CC(F)(CNC(c2cc(Cl)no2)=O)C1 24850,c1(C(N(CCC(C)NC(=O)CC2CCCCC2O)C)=O)nnn(C)c1N 24851,c1(SC)nc(N2CCC(C(=O)NCc3c(F)cccc3F)C(O)C2)cc(C)n1 24852,c12cc(C(C)(C)C)cc(C(C)(C)C)c1N2.c1(C2C(OC)CC2)ccc(C)cc1 24853,Cc1cnncc1C(=O)NC1(CC=CC(=O)NCC2CN3CCC2C3)CCC1 24854,C1(NC(c2ccncc2Br)=O)CN(C(C2CCCCO2)=O)CC(F)(F)C1 24855,C(=O)(CC(C)CCC=C(C)C)N(C)CC1N(C(C(CC)NC(C)=O)=O)CCC1 24856,c1(CNC(CCSCCC)=O)ccc(CN(C)C(c2ccncc2F)=O)cc1 24857,CS(=O)(=O)C1(C(=O)NC2CC(CNC(C34CCCN3CCC4)=O)C2)CCC1 24858,CC1CN(C(=O)C(F)(F)c2csc(=N)[nH]2)CCC1NC(=O)CN1CC2CC2C1 24859,c1(NC(=O)CC(c2ccc(F)cc2)NC(=O)CN2CCCC2)c(Br)ccnc1Cl 24860,Cc1n[nH]cc1CC(=O)NC(CO)C(C)NC(=O)CC(C)n1cccn1 24861,Cc1ncnc(C)c1CC(N1CCOC(C2CN(C(C3CNC(=O)N3)=O)C2)C1)=O 24862,C1(F)(C(=O)NCC2(NC(Cc3ccc(C(N)=O)cc3)=O)CC2)CC12CCCCC2 24863,C1(C(N2CC(C(C)C)N(C(=O)Cc3nncs3)CC2)=O)CCC(=O)C(C)C1(C)C 24864,C(=O)(CC(C)C(F)F)N1CCC(CN(C(c2ccnc(C(F)F)c2)=O)CC)CC1 24865,CCC(C)(C#N)C(=O)NCc1ccc(C(=O)NC2(CO)CC(F)(F)C2)cn1 24866,c1(C(=O)NC(CNC(=O)C(F)OC(F)(F)F)C2CC2)cc2c([nH]1)CCOC2 24867,S(=O)(=O)(c1ccc(CC(=O)NCC#CCNC(=O)CC#N)cc1)CSC 24868,Cc1cnn(C)c1CNC(=O)N(c1nnc(C(C)C)s1)C 24869,C1(NC(C2CCCCCN2C(C2CC(F)(F)C2)=O)=O)C2CCC(F)(F)C12 24870,CON=CC(=O)N1CCC(C(=O)NCC2CC2c2ccco2)O1 24871,N1(Cc2ccc(C)c(C)c2)CC2C3CCC(C2C1)N(C(=O)CC1CCCCC1)C3 24872,c1(C(=O)NC2CC(C)CN(C(c3ccc(=N)[nH]n3)=O)C2)ccc2c(c1)CCCC2 24873,CCCCC(CNC(C12CCC(C1)C2)=O)NC(c1ccsn1)=O 24874,N1(C(C2CCCSS2)=O)CC(NC(C2(C(F)F)CCC2)=O)CC2(CCC2)C1 24875,CCC(C)(CO)C(=O)N1CCCOC(CCNC(=O)CCC(=O)N(C)C(C)C)C1 24876,Cc1cccc(-n2nnc(OC3CC(F)CN3C(=O)OC(C)(C)C)c2CO)c1 24877,c1(N2CCC3(CN(C)C3)C2)ccc(Br)c(S(=O)(=O)NC2C(CO)CCC23CCC3)n1 24878,CC(C)C(C)(C(N)=O)NC(C1CC2CC2N1C(C1CC2C=CC1O2)=O)=O 24879,c1(N2CCC(NC(N3CCCCC3c3ncc[nH]3)=O)C2)ccc(Br)nc1 24880,c1(OCCC(=O)NCC2(O)CC(NC(C=CC)=O)C2)ccccc1C(C)C 24881,c1(C(N2CC(CC(C)NC(=O)CCc3nncn3C)C2)=O)cc(N)cc(O)c1 24882,c1(C(N2CC(NC(CC(C)C(F)F)=O)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 24883,c1(CC)nn(C)cc1C(=O)N(CC(CC)NC(=O)C(C)Cc1cccc(F)c1)C 24884,c1(C(N2C(CC)CCCC2)C(=O)NC2CCOC2)cc(=O)n2ccccc2n1 24885,C(c1ccc2c(c1)CCO2)=CC(=O)NC(CNC(c1c(CC)onc1C)=O)C 24886,c1(C(=O)NCC2CCN(C(C(C)=C3CCCC3)=O)C2)cccn2c(C)nnc12 24887,Cc1csc(=NCC(=O)N2CCC3CCCC23CNC(=O)C(=O)NCC2CC2)[nH]1 24888,C(=O)(C1CCCc2nc[nH]c21)NCC(CNC(c1nc(OCC)sn1)=O)(C)OC 24889,C1(C(=O)NCC2C(NC(c3nc(OC)c(C)s3)=O)C2)CCc2ncnn2C1 24890,c1(OC)cc(N2CC3CN(C(c4ccco4)=O)C3C2)nc(C)n1 24891,CC1(CNC(c2cn(CCO)nn2)=O)CCN(C(C2(N(C)C)CCC2)=O)CC1 24892,C=CCC(CNC(C1CCN(C)C1CC)=O)C(=O)N(CC(C)(C)C)CC(C)C 24893,c1(C(N2C(C3CCN(C(CCC(C)C)=O)CC3)CCC2)=O)ccc2n[nH]cc2c1 24894,N1(C(c2c(C)[nH]nc2C(F)F)=O)CC(NC(=O)C=Cc2cnc[nH]2)CC(O)C1 24895,C(=O)(C(O)CC1CC1)N(CCNC(C(C)OCC1CC1)=O)Cc1ccccc1 24896,C(CNC(=O)CCCN(C)C)(C(C)(C)C)NC(CCNC(C)=O)=O.CCSCC 24897,Cc1nn(CCF)cc1NC(c1nnnn1CCN(C)C)CC12CC(CO1)C2 24898,C(=O)(CS(=O)(=O)CCO)NCC(C1CC1)NC(C1(CC#C)CCOCC1)=O 24899,Cc1n[nH]c(C)c1C(C)C(=O)N(CC)CC1CCCN1C(=O)CC1CCOCC1 24900,c1(N(C2C3CCC2CNC3)C(c2n(C)ccc2)=O)nc(Cl)c(Br)cc1O 24901,N1(C(C=COCC)=O)CCCC(N(C)C(c2ccc(OCCF)cc2)=O)CC1 24902,C(=O)(C(CN(C)C)CC(C)C)NCC1C(C(=O)NC2(CC=C)CCCCC2)C1 24903,C1(CNC(C(C)n2cccn2)=O)CC2CC2N1C(=O)C=CCN1CCOCC1 24904,Cc1cccnc1CC(=O)NC1CC(C(=O)N(CCC#N)C2CC2)C1(C)C 24905,c1(OC)cc(F)c(CC(=O)NCCNC(c2cnc(C(F)(F)F)s2)=O)c(Cl)c1 24906,c1(C(C(=O)NCC2(F)CN(C(C3CC(OC)C3)=O)C2)(C)F)ccc(F)cc1 24907,c1(C2C(C(=O)NC3CCCC3C(F)(F)F)C2)ccccc1Br 24908,c1(C(=O)NC2CC(C)(CNC(CC=C)=O)C2)cccc(OC)c1 24909,Cc1ccc(C(=O)NCc2cc(C(=O)NCC3(O)CSC3)no2)c(C)c1 24910,c1(OCC)cc(C(=O)NC(C(=O)OCc2ccccc2)C2CC2)ccn1 24911,C#CCC(C)(C(=O)NCC(CCC)OCC)NC(=O)C(CC)C(=O)OC 24912,O=C(C1=NOCC1)N1CCC(C2CCCCN2C(c2n[nH]cc2Cl)=O)C1 24913,C(CCCCCN)N(C(=O)C(N)CC1CCS(=O)(=O)C1)C 24914,C1(NC(C(=O)NC2CC2)=O)CCCOC12CCN(C(C1(C3CC3)CCC1)=O)CC2 24915,c1(-c2cn(C3(C(=O)OC)CN(C(C4(C)CNC(=O)C4)=O)C3)nn2)cc(OC)nn1C 24916,c1(C(=O)NC(CNC(C2CN(C)C(=O)N2)=O)CO)c(F)ccc2[nH]ccc12 24917,c1(CNC(c2cc(=O)cc[nH]2)=O)cccc(NC(C2OCCCO2)=O)c1 24918,c1(C(N(CC(CC)NC(C2C3CC(=O)CC23)=O)C)=O)nc(C)oc1C 24919,C(C(=O)N(CC(=O)NCc1nonc1C)CC(C)C)(C(C)C)SCC 24920,c1(OC)ccccc1OC(C)C(=O)NCCC(C)N(C)C(c1c[nH]c(C#N)c1)=O 24921,C1(OCC(=O)OC)CCN(C(C2CN(C(c3ocnc3C)=O)CCS2)=O)CC1 24922,C#CC1(O)CC(C(N2CC(F)CC2C(=O)N(CC=C)CCC)=O)C1 24923,C12(C(N3CC(CC)(CC)C3)=O)CCCC1CCN2C(=O)CCC1OCCO1 24924,CN1CCC(CC(=O)NC(C)(CNC(=O)CN(C2CCC2)C)C2CCC2)CC1 24925,N1(C(C2CC23CCCC3)=O)CC2CCC1C(CNc1cc(F)ncn1)C2 24926,C1(NC(c2cc(CC)nn2C)=O)CC2CC1N(C(c1cnn(C)c1C)=O)C2 24927,CCC(C(=O)N1CC(CCNC(c2ccn(C)c2C)=O)C(C)C1)C(C)C 24928,Cc1cc(C(N2C3CC2CN(C(c2c(O)cccc2O)=O)C3)=O)cc(Br)c1 24929,Cc1ccc2cc(C(=O)N(CCNC(=O)Cc3ccc(C)s3)C(C)C)cnc2c1 24930,c1(C(=O)NC2(C)CCC(NC(c3ccn(C)n3)=O)CC2)ccc2c(c1F)CCC2 24931,Cc1ccc(NNC(=O)c2csc3cc(Br)ccc23)cn1 24932,c1(OC)cc(C=CC(N2CCC(NC(=O)C(F)CC3CCCC3)C2)=O)sn1 24933,c1(C(=O)NC2CCN(Cc3cc(F)ccc3Br)CC2)ccc2c(c1)CNC2 24934,N#Cc1ccc(Cl)c(C(=O)NCCNC(C2CCOC2c2ccccc2)=O)c1 24935,c1(COC)n[nH]c(=NC2(CNC(=O)CCc3c(N)cnn3C)CCCCC2)s1 24936,O=C(C(Cc1ccccc1)NC(=O)C1CC1)Nc1nnc(Cc2ccccc2)s1 24937,C1(NC(CCCSC)=O)CCC2CCN(C(=O)C=Cc3cncn3C)C1C2 24938,c1(C(=O)NCC2C3CN(Cc4cccc(C)c4Br)CC32)ccc2scnc2c1 24939,C1(NC(c2ccc(C(=O)OCC)o2)C)CCC(CC(C)(C)C)C1 24940,Cn1nc(C(N2CC(CCNC(c3cnoc3C3CCC3)=O)C2)=O)cc1Cl 24941,CC1CC2(C(N3CC(SC(F)(F)CF)C3)=O)CC12 24942,C1(C(=O)NC2(CC(=O)NCC(CNC(N)=O)O)CC2)CC=CCO1 24943,c1(C(=O)NC(CN(C(c2ccc(F)c(O)c2)=O)CC)C)ccc(C)cc1OC 24944,N1(C(c2ccc(SC)cc2)=O)CCC(NC(=O)CN2C(=O)COCC2=O)C1(C)C 24945,CC(CC(=O)N1CCC(N(CC(C)C)C(C2CCC(O)C2)=O)CC1)C(F)(F)F 24946,C=CC(CC)CC(=O)NCC(C(=O)NCc1ccc(C(N)=O)o1)C(C)C 24947,c1(C(N2CC(O)(C(C)NC(CCC(=C)C)=O)C2)=O)nc(Cl)ccc1Cl 24948,c1(OCC)ccc(CN(C2CCC2(F)F)Cc2ccccn2)c(C)c1 24949,N1(C(c2ccc(OC)c(C)c2NC2COC2)C=O)CCCC(C2CCC2)CC1 24950,c1(CN2CCC(NC(C(c3ccnn3C)C)=O)C(O)C2)ccc(F)c(C#N)c1 24951,C12(C(N(C3CCCC(NC(c4coc(C5CC5)n4)=O)C3)C)=O)CCC(CC1)C2 24952,C(C(=O)NCCCC(C)NC(=O)CNC(c1cccnc1)=O)(C(C)(C)C)SC 24953,Nc1nc(NC(=O)NCCS(=O)(=O)Nc2c(Cl)nsc2Cl)ccc1O 24954,C=CC(C)(O)CC(=O)N1CCC(C(C)(C)C(=O)NC2CCOC2C)C1 24955,N1(C(c2c(C)non2)=O)CCC(C)(C(N2CCC(CN(C)C)C2)=O)C1 24956,CC(O)C(C)C(=O)NC1(CNC(=O)CCCc2cccs2)CC1 24957,N1(C(C2N(CCC)C(=O)CC2)=O)C2CCC1CN(C(C1C(C)(C)C1(F)F)=O)C2 24958,C(=O)(CCCCC#N)NCC1CN(C(COCCC=C)=O)C(C)C1 24959,C1(NC(CCN(C)CC)=O)CC2CC(C1)N(C(=O)Cc1ccccc1Cl)C2 24960,c1(OC)nc(Cl)ccc1C(N1CCCCC(NC(C2CCN(C)C(C)C2)=O)C1)=O 24961,C(=O)(C1=CCC(C)(C)CC1)NC1(CCCCNC(c2cc(C)sc2C)=O)CC1 24962,C(=O)(CCCC(N)=O)N1CCC(NC(C2C(C)C2(F)F)=O)C1C1CC1 24963,CCN=c1[nH]cc(C(=O)NCC2CCN2C(c2cn(C3CCC3O)nn2)=O)s1 24964,CCC(C)(COC)C(=O)NC1C=CCC(C(=O)NCC(C)C(C)O)C1 24965,C1(C)(C(=O)NCC(C2CCCCC2)NC(C(C(C)C)CO)=O)CC2CCC(C1)S2 24966,N1(C(C2CCN(c3ccccc3)C2)=O)CCc2sccc2C1c1ccc(Cl)cc1 24967,c1(NC2CCC(N(C(=O)CN3CCC(O)CC3)C)CC2)ncnc2[nH]ccc12 24968,Cc1cnc(C(N2CC3CC2C3C(=O)N(C)C(C2CCC2)C)=O)c(F)c1 24969,c1(OC)ccc(C)cc1C(=O)NCCCN(CCO)C(C1CCC1C(=O)OC)=O 24970,c1(NCC)ccc(Cl)cc1C(N1CCC1CNC(c1cccnc1C)=O)=O 24971,N1(C(CC(CNC(=O)Cn2cc(C)cn2)OC)=O)CCC(C)(C)C1C 24972,c1(C(N2CCN(CC#CCC)CC2)C(=O)NCCOC)ccc(OC)c(OC)c1 24973,Cc1cccc(C(CNC(C2CN(C)C(=O)N2)=O)NC(=O)Cn2cnc(=N)[nH]2)c1 24974,N1(C(c2n[nH]c(C)c2C)=O)CC(C)(C(=O)NCC(c2ccccc2)O)CC1(C)C 24975,C1(C(N2CCC(C3N(C(CCC(=C)Cl)=O)CCC3)C2)=O)CCc2cnc(C)n2C1 24976,C=C=CC(C)C(=O)NC1(C(F)F)CC(NC(=O)CCCOCCOC)C1 24977,N1(C(c2cccc3ncoc23)=O)CC2CCCC(N=c3[nH]nco3)C2C1 24978,CCC(CCCC(=O)N1CC2COCC2O1)NC(C1(F)C(C)(C)C1(C)C)=O 24979,N1(C(CCC(C)OCC)=O)CCN(C(=O)C(C)n2ccnn2)CC1C(C)C 24980,CC1CCN(C(c2cc(Cl)c(Cl)[nH]2)=O)CC1NC(=O)Cn1ccc([N+](=O)[O-])n1 24981,N1(C(C(=O)NC(C(=O)OC)C)c2ccoc2)CC(c2cccc(Cl)c2)OCC1C 24982,CCCCC(C)C(=O)NCCn1cc(CNC(=O)CSc2ccc(Cl)cc2)nn1 24983,c1(C(N(C(CCNC(C=NOC)=O)C)C)=O)cccc2c(C)coc12 24984,C=CC(CCC)CC(=O)NCc1ccoc1C(=O)NC1(C)CC1(C)C 24985,C1(NC(C2CC(=C)C2)=O)CC2CCC1CN(C(c1cn(C3CCOC3)cn1)=O)C2 24986,C(=O)(CCC(C)(C)O)NC(C(C)C)CNC(=O)Cc1ccc(C(N)=O)cc1 24987,C1(COC)(NC(=O)CCNC(N)=O)CCN(C(C2CC3(CSC3)C2)=O)C1 24988,N1(C(C(CC(F)F)NC(c2c(C)ncs2)=O)=O)CC2C3CCC(C3)C12 24989,C1(C(=O)NC(C(=O)NCC(C)(C)SC)(C)C2CCC2)Cc2ccccc2C1 24990,c1(C(N(C2CCN(C(=O)CCc3ncco3)CC2)C)=O)ccc(F)c2c1OCC2 24991,O=C(C(F)CC1CCOCC1)NCC(F)(F)Cn1cc(CCN2CCSCC2)nn1 24992,Cc1cc(C(N2CC3CN(Cc4ccnc(Cl)c4C)CC3C2)=O)c(C)cc1O 24993,C1(C(C)C)CCCCC1CNC(N1CC(C(C)(C)S(C)(=O)=O)C1)=O 24994,CCC(CNC(=O)C(C)(C)c1ccccc1)(CC)NC(=O)CN(C1CCSC1)C 24995,C1(CC)CN(C)CCCN1C(=O)C(CC(N)=O)NC(=O)C(C(C)OC)N(C)C 24996,c1(NC(C2CCN(c3ccnc(Br)n3)CC2)=O)ccc2c(c1)C(=O)CCC2 24997,c1(OCC=C)ccc(CN(CCCC)C(C)=O)cc1.C1(=O)C(CC)N1 24998,C1(OC(c2ccccc2)C(C)C)CC(C(=O)NC2CC3CNC2C3)CCC1O 24999,Cc1cc(CNC(=O)C(CC2CCCC2)NC(=O)C(C)C#N)no1 25000,c1(CN2C(CCP(C)(C)=O)CCCC2)ccc(Cl)c(Br)c1 25001,CC1(CNC(c2cc[nH]n2)=O)CCCN1C(=O)C=CCO 25002,C=CC1(C(=O)NCc2ocnc2C(=O)NCC2CC(N(C)C)C2)CCOCC1 25003,c1(C(N(CC(C)CNC(=O)CCCn2ccccc2=O)C)=O)cc(Cl)ccc1N 25004,CCCC(C)C(=O)NC1CC(F)(C(=O)NC2(O)CN(C(=O)OC(C)(C)C)C2)C1 25005,C1(C(N2CC(CO)(CO)C2)=O)CCC(CNC(c2n[nH]cc2C(F)(F)F)=O)CC1 25006,n1(CC)cnnc1CNC(=O)C(C1CC1)N(C(=O)Cc1nonc1C)C 25007,N1(CCC)CC(C(=O)NC(C)(C)C(C)NC(=O)C(c2ccc(F)cc2)=O)CC1=O 25008,C1(NC(CCCCCSC)=O)CC2(CCN(C(c3cc4n(c3)CCC4)=O)CC2)C1 25009,c1(CCC)ccc(N)c(C(=O)NCC=CCNC(=O)C=CC2CCC2)c1 25010,C1(C(=O)OCC)CN(C(=O)C(Br)=CCF)CC1C1CC1 25011,N1(C(CCNC(=O)OC)=O)CC2C3CCC(C2C1)N(C(=O)C(C)(C)F)C3 25012,C=CCC(CC=C)C(=O)NC(CN(C)C)C(=O)NCC(=O)OCC 25013,C1(CNC(c2c(C)cnn2C)=O)CN(C(c2occ(C)c2C)=O)CC12CC2 25014,C(CC(C)C(=O)N1CCC(C(O)CNC(c2cccn2C(C)C)=O)CC1)OC 25015,C=CCCCCC(=O)NC1CCCN(C(c2cc(OC)ncc2F)=O)C1C 25016,N1(C(c2cc(C)n(C3CC3)n2)=O)CC(CN(C)C(c2cscc2F)=O)C2(CC2)C1 25017,N1(C(C(COC(C)(C)C)(C)C)=O)CC2CC(NC(=O)CCC3CCOC3)C1C2 25018,c1(C(=O)NC(C2CC2C(N2CCCC(O)C2)=O)C)ccccc1O 25019,N1(C(C2C(C(=O)OC)C2)=O)CC2CCN(C(C3CCc4n[nH]cc4C3)=O)C2C1C 25020,C1(NC(CCn2ccc(C)n2)=O)CS(=O)(=O)CC1NC(c1cnc(S)[nH]1)=O 25021,c1(C(N2CCC(NC(C3CCCCS3)=O)C23CCC3)=O)noc2c(F)cccc12 25022,C(=O)(C(C)(C)CN1CCOCC1)NCC(CNC(C1(n2nccn2)CC1)=O)OC 25023,Cc1ccnc2sc(C(=O)N(CC(=O)O)C(c3cn(CCN(C)C)nn3)C)c(C)c12 25024,CC1CN(c2nnnn2CCCC(C)(C)C)C(C)C1C 25025,C(=O)(CCNC(=O)C(c1cnsc1)N(CCCN(C)C1CC1)CCOC)OCC 25026,C12(C(=O)NCC3C(NC(CN(CC)CC)=O)CCCC3)CCCN(CC1)C2 25027,CC(C)CC(CNC(C1OCCC1C(C)C)=O)C(=O)Nc1ccccc1N=[N+]=[N-] 25028,c1(CC)onc(C(N2CCOC(C(=O)N(CC(C)CO)C)C2)=O)c1C 25029,C1(NC(c2n(C)c(S)nc2)=O)CN(C(c2noc3c2CCCC3)=O)CCC1(C)C 25030,C(C(O)CC(=O)NC1CC1CC(C)(C)C)NC(C(C)(C)NC(C)=O)=O 25031,CN1CCC(N=c2[nH]c(=NCC3(C)CC4(CC4)C3)[nH]c3c2SCC3)C1 25032,C(c1c(C)nn(C)c1Cl)=CC(=O)NC1C(OC)CN(C(c2cc(=O)cc[nH]2)=O)C1 25033,C1(NC(C(C2CC2)OC)=O)CCN(C(c2cn(CC(=O)N(C)C)nn2)=O)C1C1CC1 25034,C(C(c1ccccc1)NC(=O)CCF)(C(C)C)NC(c1c(OC)nsc1)=O 25035,C(C(=O)NCC1CC(NC(c2csc(CO)n2)=O)C1)(C(C)O)NC(C)=O 25036,C1(NC(CC2CC(=C)C2)=O)C2CC3CN(C(c4n[nH]c5c4CCCC5)=O)C1C3C2 25037,c1(N(C2CNCC2F)C(c2ccc(OC)nc2OC)=O)ncnc2c1ccn2C 25038,C(=O)(C1=Cc2cc(Br)ccc2OC1)NC1CCN(C(C)=O)CCC1(F)F 25039,c1(C(N2CCC3(C(C(=O)Nc4ncc(Br)s4)C3)CC2)=O)c(F)c(F)cc(F)c1F 25040,c1(OC(C)C)ccc(CC(=O)N(C2CC2)CC2(C(F)(F)F)CCCOC2)cc1 25041,CCC(C)(CC)NC(C1CC(CCNC(=O)CC(=O)N(C)C)C1)=O 25042,C1(N)CCCCN(C(C)(C)C)C1.C1(CCC(=O)NC)CCC(C(=O)OC)N1C(C)(C)C 25043,C1(C(N(C)Cc2ccc(OC)c(F)c2)=O)CC12CCN(c1ncccc1F)CC2 25044,C(=O)(C(C)CS(=O)(=O)NC1CCC(CC(C)(C)C)C1)OC 25045,CCC(c1ccccc1)=CC(N1CCC(C)C1CNC(c1c(C)coc1C)=O)=O 25046,C1(CNC(CCN(CC#C)C(C2CC(C)CO2)=O)=O)CCCOCC1 25047,c1(C(=O)OCc2ccc(CC=C)cc2)cc(C)c(Br)c(Cl)c1 25048,N1(C(C2(OC)CCN(C(c3c[nH]c(=O)cn3)=O)C2)=O)CCCCC(CO)C1 25049,N1(C(Cc2cc(C)[nH]n2)=O)CCC2(CCN(C(c3cc(Cl)c(N)c(Cl)c3)=O)C2)C1 25050,C1(C(=O)NCCCN(C(c2c(N)cccc2Cl)=O)CC)CCn2c(cnc2C)C1 25051,C(N=c1cc[nH]cc1)C1CCN(C(=O)Nc2c(C)n(-c3ccccc3)nn2)CC1 25052,C=CC(O)C(=O)N1CCC(n2cc(CNC(=O)COCCCC)nn2)C1 25053,C1(NC(c2ccsn2)=O)COCCN(C(=O)CCc2ccsc2)C1 25054,c1(C(N2CCOC(CN(C)C)C2)C(=O)NCCCCCC)cc(F)cc(Br)c1 25055,C(=O)(C1SCc2cccnc21)NCC=CCNC(c1cc(CCC)[nH]n1)=O 25056,C(=O)(C1CCc2c(F)cccc21)NCc1cc(OC)ns1 25057,C1(C(=O)NC2C(C(N(C(C=C)C3CC3)C)=O)OCC2)CCOC(C)C1 25058,C(=O)(C(C)(C)CNC(=O)CCCOC(C)C)NCC(C1CC1)OCC 25059,c1(OC)cccc(CC(=O)OCC2CC(C)N(C(=O)C=Cc3cocn3)C2)n1 25060,c1(OC)cc(I)c(NC(C2CC2NC(=O)Cc2ccc(Br)cc2I)=O)cc1OC 25061,c1(CCCNC(=O)COCCNC(=O)CCc2cnco2)nncs1 25062,N1(C(C2C(C)(C)C2(F)F)=O)CCC(CNC(=O)Cn2ncc(O)nc2=O)C(O)C1 25063,N1(CCC(=O)NC(CN(C(c2ccncc2)=O)CC)C)CCCCCC1 25064,c1(C(=O)NC2C(C)(C)N(C(=O)CCCC#N)CC2)ccc([N+](=O)[O-])cc1Cl 25065,C=CCC(C(=O)NCC(CCOC)NC(c1[nH]nc2ncccc12)=O)C(C)C 25066,c1(C(=O)NC2CC(NC(CS(CC)=O)=O)C2)cc(O)nc2cc(F)ccc12 25067,C1(C(N(CCC(C)NC(=O)CN2CCCC2C)C)=O)COCCOC1 25068,C(C(=O)OCC)(C(C)C)NC(N1CCCC(c2c(C(=O)OCC)cn(C)n2)C1)=O 25069,C1(O)(CCNC(C(C)c2ccco2)=O)CN(C(=O)CCSCC(N)=O)C1 25070,c1(C(N2CC(O)(CNC(c3ncn(C(C)(C)C)c3)=O)C2)=O)ccc2c(c1)COC2 25071,C1(CN)CS(=O)(=O)C2CN(C(c3c(OC)c(F)c(Br)cc3)=O)CC12 25072,CC1(CO)CCCN1C(C1CCC(NC(=O)CCC2CC2(F)F)C1)=O 25073,C1(C(=O)N(C2CN(C(C)C)C2)C)(CC)CCN(C(=O)C(C)(CO)NC(C)=O)C1 25074,Cc1cc[nH]c(=N)c1C(=O)NC(CNC(=O)C(C)c1cccs1)C1CC1 25075,c1(OC)ccc([N+](=O)[O-])c(C(N2CC(F)CC2C(=O)NCC2CCOC2)=O)c1 25076,C1(C(=O)NC(C(=O)N(C)CC)C)COCCN(C(c2c(C)nn(C)c2N)=O)C1 25077,S(=O)(=O)(c1cc(C)ccc1C)N(CC(CC)CC(C)C)C1CCNCC12CC2 25078,c1(OC)ncc(C(N2CCCCC2C2CCN(C(=O)C(C)SC)CC2)=O)cc1F 25079,c1(OC)cc(OC)cc(C(N2CCNC(C(=O)OC(C)C)C2)=O)c1.C1(=O)CN1 25080,c1(C(=O)NC(CNC(C(C(C)C)(C)O)=O)CO)coc(S(N)(=O)=O)c1 25081,CCCCC(CC)C(=O)N1CCCC(NC(c2ccc(OC)nc2C)=O)CC1 25082,C1(OCC)CN(C(=O)C(=Cc2c[nH]cn2)F)CC1CNC(c1cn(C)nc1Cl)=O 25083,c1(C(N2CCCC(NC(C3CC3(F)F)=O)C2)=O)c(OC(F)F)cccc1Br 25084,c1(CCC(N2CC(C)(NC(c3c(OCC)scc3)=O)C2)=O)n[nH]c2ccccc12 25085,Cc1cc(C(=O)NCC2CCCC2C(N2CCCC(C#N)C2)=O)cc(O)n1 25086,c1(NC(CCC(C)C)=O)ccc2c(c1)CCN(C(c1cccc3nscc13)=O)C2 25087,CC(C)(C)C(C(=O)N1CCC(NC(=O)CC2CCC3CC23)CC1)N1CCOC1=O 25088,Cc1cccn(CC(N2CCN(C(=O)CCCCCN(C)C)CC2C)=O)c1=O 25089,N1(C(CCCOCCC)=O)CCC2CCCC12C(=O)NCCCC1(O)CCC1 25090,c1(NC(=O)C(O)CCCc2ccc3ccccc3c2)ccc2ccccc2c1O 25091,c1(CC)cc(C(=O)NCCCN2CCN(C(=O)C=CC(C)C)CC2)cn(C)c1=O 25092,N1(C(C2(C3CC3)CN(C(CC3N(C)CCCC3)=O)C2)=O)CCCC2C(O)CC12 25093,N1(c2ccnc(NCCS(CC)=O)n2)CC(C)(C)C(F)(F)C1 25094,c1(C(=O)NC(CCC)C(N2CC(O)CC(C)(C)C2)=O)ccc(C#N)c(C)c1 25095,C1(NC(C(C)C(C)O)=O)CC2CCCC(C1)C2NC(=O)Cn1ccc(O)nc1=O 25096,C(CCCC(C)(C)C(=O)NNC(=O)C1CSC1)NC(c1cc(C)c(F)c(C)c1)=O 25097,Cc1nc(=N)[nH]c(C)c1C(N1CC(NC(c2ccc(C(C)C)cn2)=O)C(C)C1)=O 25098,c1(C(=O)NC2C(NC(C3(C(C)(C)C)CCCC3)=O)C2)cccc(CCO)c1 25099,C(=O)(CC(C)C(F)(F)F)N1C(C(N2C(COC)COCC2)=O)CC2CC21 25100,C1(F)(CNC(C(C2CCC(=O)N2)C)=O)CCN(C(=O)CC2SC(=N)NC2=O)CC1 25101,N1(C(C2CCCC(C(N)=O)C2)=O)CCCC(C)(CNC(c2ccc(CO)s2)=O)C1 25102,N1(C(CSCCN(C)C)=O)CCCCC(N=c2ccc(C(F)(F)F)n[nH]2)C1 25103,NS(=O)(=O)CC(=O)NC1CN(C(c2cccc(C3(O)COC3)c2)=O)C2CC12 25104,c1(-c2nc(NCCCC(c3cc(C)sc3C)=O)sc2)cn(C)c(=O)nc1O 25105,N1(C(C(C=C)O)=O)CC(C2CCCN(C(c3ccc([N+](=O)[O-])cc3F)=O)C2)C1 25106,Cc1ccc(C)c(C(C)N(C)Cc2cc(-c3ccccc3)[nH]n2)c1 25107,c1(C(=O)NCCN(C)C(C2CCc3ccnn3C2)=O)cncc2ccsc12 25108,C1(NC(c2cnn(-c3ccncc3)c2)=O)CN(C(=O)C=CBr)C2(CCC2)C1 25109,C(=O)(CC(C)(C)CC(=O)NCC1(C2CC2)CCN(C(=O)Cc2ccsc2)C1)OC 25110,C(=O)(C1=NOC2(CCC2)C1)N1C(CNC(c2occc2Cl)=O)CC(O)C1 25111,C(=O)(C(F)CCC(C)C)NC(CC(=C)C)C(=O)NC(c1cccnc1)CC 25112,N1(C(C(c2n(C)cnc2)O)=O)CCCC(CCC(=O)N(CCC(C)(C)C)CCO)C1 25113,C(=O)(C1CCCCc2ccccc21)N1CC(O)(C(C)NC(CCCOC)=O)C1 25114,c1(C(C)C)cc(C(=O)NC2CCC(NC(c3ccc(Cl)c(N)c3)=O)C2)cc(O)n1 25115,NS(=O)(=O)CC(=O)NCC1(F)CN(C(=O)CC(F)(F)F)C1 25116,c1(C(N2C(CNC(C(C(CC)C)O)=O)CC2)=O)ccc2nc(COC)[nH]c2c1 25117,c1(CC)[nH]nc(C(=O)NC(CCC2CCC2)C(=O)NC(c2cnc(C)s2)C)c1C 25118,N1(C(C=CCOC)=O)CC2OCC(NC(=O)CCSCc3ccccc3)C2C1 25119,CC(c1cccnc1)=CC(=O)NCC1CC2CCC1N2C(=O)Cc1ccco1 25120,c1(C(=O)NCCN(C(=O)C(=O)NOC)CCC)ccnc(OC(C)(C)C)c1 25121,c1(C(N2CCC(NC(Cc3c(C)ocn3)=O)C2)=O)cc(O)cc(Br)c1 25122,CC(CC(=O)NCC1C(C(=O)NC(CC(N)=O)C2CC2)C1(C)C)C(F)F 25123,CCCC(CC1CCCC1)C(=O)NCC1CCN(CC(O)COC)CC1 25124,c1(OC)cc(F)c(F)cc1C(N1CCC(C)(C(=O)O)CC1)=O 25125,c1(OC)ccc(C(=O)N(C)CCNC2CC2)cc1S(=O)(=O)NC(=O)C(C)S(N)(=O)=O 25126,C(=O)(C(C(C)(C)C)NC(=O)C(C)C)NCCC1(NC(CCC(C)OC)=O)CCC1 25127,C(=O)(C(C)(C)C(O)CC)N1C2C(NC(c3cccc(CC)c3)=O)CC(C2)C1 25128,c1(C(N(CCNC(c2cc3ccccn3n2)=O)CC)=O)ccc([N+](=O)[O-])cc1Cl 25129,C1(CNC(C2(CC#C)CCC2)=O)CCCN(C(=O)C=CC2CCOCC2)CC1 25130,CCCC(C(=O)NC1CCCN(C(c2ccc(F)c(C(F)F)c2)=O)C1C)C(C)C 25131,Cc1nn(C2CC2)c(C)c1C(=O)NCC(C)(C)OCCNC(=O)CCC1(C)CC1 25132,CC1CCC(NC(c2ccc(C#N)n2C)=O)CN1C(c1cnc(C2CC2)nc1)=O 25133,C1(CNC(c2c(C)coc2C)=O)CC2(CCN(C(C3(O)CC(C)(C)C3)=O)CC2)C1 25134,N1(C(CCC(=C)C)=O)CCCC(CO)(NC(=O)CCSc2ccc(C#N)cc2)C1 25135,C1(NC(c2cnc(C3CC3)nc2)C)CC2(C1)CN(c1ncncc1I)C2 25136,CC1(C)C(C(N2CC(CNC(=O)C(c3ccccc3)O)C2)=O)CCS1(=O)=O 25137,c1(C(C2(OC)CCOC2)NC(CCC)C2CCCC2)nnnn1CCC1CC1 25138,CC1CN(C(C2CCCC(F)(F)CC2)=O)CC(C)CN1C(c1cnccc1Cl)=O 25139,C1(C(=O)NC23CC(C(N4C(CCOC)CCCC4)=O)(C2)C3)CC2CC1CC2O 25140,c1(C(N2CCCC(CCNC(C(COC)O)=O)C2)=O)cc(C)cc(Cl)c1 25141,C1=C(CNc2nc(C3CC3)co2)CCC1 25142,C1(C(=O)NC(C2CCN(C(CC(C)C)=O)C2)C)Cc2ccccc2N1C 25143,c1(OCC)ccc(C2(C(=O)NCC3C=CCN3C(=O)CC(C)OC)CCC2)cc1 25144,c1(C(=O)NC(C2CCCN2C(=O)Cc2ccc(Cl)s2)C)csc(-c2nc[nH]n2)n1 25145,c1(-c2ccc(CN(C(CCC)C)Cc3ccncc3)s2)c(F)cccc1Cl 25146,c1(OC)cnc(F)c(C(=O)N(C(C)CNC(c2cncc(C(=O)N(C)C)c2)=O)C)c1 25147,S(=O)(=O)(c1cnn(C)c1)N1C(C(=O)NC(C(=O)OC)C(C)O)CC2CC21 25148,CCC(C)CC(=O)C(=O)NC(C)(C)C(=O)NC(C1CSC1)C 25149,CC1(C)CCCOC1C(=O)NCCCC(=O)NCc1cccc(O)n1 25150,N1(S(CC)(=O)=O)CCCCC(NCC2CCCC2OCCN2CCN(C)CC2)C1 25151,C12(C(N3CC(C)(COC)C3)=O)CCN(C(=O)C(C3CCCCC3)C)CCC1C2 25152,C1(CCNC(CCCOCCOC)=O)CCCN(C(=O)Cn2cnnc2)CC1 25153,CC(C(=O)N1CCC(N(C)C(C2CCCN2CC(F)(F)F)=O)CC1)C(F)(F)F 25154,N1(C(C2CC2(F)F)=O)CC2CCC1C1CN(Cc3ccnc(C(F)(F)F)c3)CC21 25155,CCCCCCCC(=O)NC1C(C)CCN(C(=O)COc2ccc(O)cc2)C1C 25156,CC1CCN2N=C(C(=O)NCCN(C(=O)C(C)NC(N)=O)C3CC3)NC2=N1 25157,c1(C(=O)NCCCCNC(c2cncc(OC)c2)=O)cc(C)c2c(c1)CCCN2 25158,C12=CC=C(C=C1)C2NC(c1n(CCC)nnn1)c1cc(COC)no1.C(C)SC 25159,N1(C(CN(C(=O)CCC2CC(C)C2)CC)=O)CC(CO)OCC1C 25160,C1(CNC(CC=C(C)C)=O)CN(C(=O)C(C2CCCCCC2)C)CC12CCC2 25161,C(=O)(CC(C)CC(C)(C)C)NCC1=CCN(C(c2c(NC(C)=O)cccn2)=O)CC1 25162,C(CC)(C(=O)NC1(C)CC(NC(=O)C(n2cc(Br)cn2)C)C1)=CC 25163,Cc1noc(C(F)F)c1C(N1CCC(CN(C(=O)CC2CCNC(=O)C2)C)C1)=O 25164,N1(CCC(C)SC)CCCC(NC(=O)C(C)C)CC1 25165,c1(NC(CCN(C(C(COC)OC)=O)CCO)=O)ccncc1F.C(C)(C)(C)N 25166,N1(C(C(C)n2cnnn2)=O)CC2CCCC(C1)N2C(c1cnc(F)c(F)c1)=O 25167,c1(CN=c2scc(CNC3(CO)C(C)(C)CCC3)[nH]2)n[nH]c2c1CCCC2 25168,c1(C(=O)NCCC(=C)CNC(=O)C(C)CC2CC2)ccc(Cl)c(N2CCNC2=O)c1 25169,C1(=CC(=O)NC(C)C(C)NC(=O)CCC23CCC(CC2)C3)CN2CCC1CC2 25170,CC1CCN(C(C2(O)CC2)=O)CC1NC(c1coc(-c2ccccc2)n1)=O 25171,C#CCCC(O)C(=O)NCC(c1ccccc1)N(C(=O)Cc1sc(C)nc1C)C 25172,Cc1scc(CNC(=O)C(C2(O)CN(C(c3nnsc3C)=O)C2)F)c1C 25173,c1(OC)ncc(C(=O)N(C(C)CNC(=O)C(O)C2CC2)C)c(C)n1 25174,O=S(=O)(c1cnn2ccc(=NCCN3CC4CC4C3)[nH]c12)N1CC(CF)C1 25175,C(=O)(N=S1(=O)CCc2ccccc21)C1C(C)=CCC=C1 25176,c1(CNC(c2nc(C)oc2C)=O)cc2n(n1)CCN(C(=O)CC1CCC1)C2 25177,CCCC(C(=O)N1CC(O)(C(C)NC(=O)C(=O)N=S(C)(C)=O)C1)S(N)(=O)=O 25178,CC(CC(F)(F)F)C(=O)NC(C)(C)CC(N1CCC(F)(CO)CC1)=O 25179,CC1CC(C(N2CC(CCNC(c3ccc(=N)[nH]c3)=O)C2)=O)CC(C)C1 25180,CCC(C(=O)N1CC(CNC(=O)CC2CCOC2=O)C1)N(C)C 25181,N1(C(c2c(C)cco2)=O)CC(CNC(C2CCC(C(N)=O)C2)=O)OC(C)(C)C1 25182,N1(C(C2(OC)CCCC2)=O)C2CCCC1CC(NC(=O)C(C1CC1)SC)C2 25183,Cc1[nH]nc2cc(C(N3CC4CC3CN4C(C3CCS3(=O)=O)=O)=O)ccc12 25184,C1(C2CC2)(OC)CN(C(=O)CC2CN(C(=O)CCCN=[N+]=[N-])C(C)(C)C2)C1 25185,CC1CCN(CC2CCN(C(=O)OC(C)(C)C)C(C)C2)CC1C 25186,C1(C)(N(C(=O)CC2CC(C)(C)CN2C(=O)OC(C)(C)C)C)CC(F)(F)C1(F)F 25187,C=CC(C)(C)CC(=O)N1C(C)CCCC1C.C1C(O)CN(C)CCN1C 25188,N1(C(C(C(=O)OCC)OC)=O)CC2CCCC2C1C(=O)NC1(C(=O)N(C)OC)CC1 25189,C1(C(N2CCC(N(C(CCc3nc(C)sc3)=O)CCO)C2)=O)COCCOC1 25190,C(=O)(C(C)CC(N)=O)N1CCC(C(=O)N(C)CCc2nccs2)(CC)C1 25191,c1(C(C)(C)C)ccc(SCC(=O)NCC(O)CNC(C2(C)C=CCC2)=O)cc1 25192,C(=O)(CC(C)C(F)F)N1CC(OC)C(NC(=O)Cc2ccc(F)c(F)c2)C1 25193,C(CC(C)N=c1[nH]c(N2CCC(CCn3ccnc3)CC2)nc2c1CC(C)CC2)SC 25194,C=C(C)C1CN(C(C2CCC3(CC3)N2C(=O)C(O)C(C)(C)CC)=O)CCO1 25195,N#Cc1cc(-c2cnn3c2OCC2(CC2)C3)cc(S(N)(=O)=O)c1 25196,C(c1ccc(F)c(F)c1)=CC(=O)NCCCCC(C)NC(=O)C(C)CC1CCC1 25197,Cc1nc(C(=O)N(CC(C)NC(=O)C(C)(C)CF)C)ccc1[N+](=O)[O-] 25198,N1(C(CC(C)n2ccnc2)=O)CCSCC1C 25199,Cn1ncc2ncc(C(N3CC4CCC3CN4C(=O)CC3CC=CCC3)=O)cc12 25200,c1(C(N2CC(NC(C(C)Cc3ccco3)=O)C2)C2CCCC2)cccc(Cl)c1Cl 25201,C(=O)(CCCCN(C)C(c1cnnn1C)=O)N(CCN=[N+]=[N-])C 25202,Cc1cc(O)cc(C)c1C(=O)NC(C)CCNC(=O)C(N1CCC(O)CC1)C 25203,C1(C(=O)NCC(CNC(C(C=C)OC)=O)(C)OC)CN(C)CC(C)O1 25204,C(=O)(C(CCCC#N)N1CC(=O)N(CCOC)C(=O)C1)NCCOC 25205,Cn1ncc(Cl)c1C(=O)NCCC1CCCN1C(C1CN(C2CCOCC2)C1)=O 25206,C1(C)(C(C)C)CCN(C(C2CCCC2NC(=O)CC(C)N(C)C)=O)CC1 25207,N1(C(C(C(C)C)O)=O)CC2(COC(CNC(C3C4CCC(C4)C3(C)C)=O)C2)C1 25208,C(CC(C(=O)NC1(C(=O)OC)CCC1)NC(=O)CC1C(C(=O)O)CC1O)SC 25209,CC1CC(CNC(c2ccc(=N)[nH]c2)=O)CN1C(=O)CCN1CCCC1 25210,C(CCOCc1nc(C(F)(F)F)cs1)(C(=O)O)NC(C(C)C)=O 25211,C1(OC)(CNC(C23CCN(CC2)C3)=O)CCN(C(=O)CN2CCC(C)C2)C1 25212,C(C)(C(=O)N1CC(C(C)NC(c2coc(C(F)F)n2)=O)C1)(C(C)C)OC 25213,C(=O)(C(C(C)(C)C)c1cccc(C)c1)N(CC(C)NC(CCC(=C)Br)=O)C 25214,C(C(CC(=O)NC1CCC(=O)NC1)NC(c1cc(OC)n[nH]1)=O)OC 25215,CC(=O)CCC(=O)NC(CC1CCC1)C(N1CCC(F)(CF)C1)=O 25216,c1(C(N)=O)ccc(=NCCCNC(C2CCN(C(c3ccns3)=O)CC2)=O)[nH]c1 25217,c1(C(N2CCCC(c3cc[nH]n3)C2)C(=O)NCC=C)cc(OC)c(OC)cc1F 25218,C1(C(=O)NC2(CC(=O)NCC3CC(OC)C3)COC2)CC(C)(O)C1 25219,CON(CCO)C(=O)CC(C(F)F)NC(=O)CC1CCOCC1 25220,C1(C(=O)NCC(CNC(C(N2CCC(O)CC2)C)=O)O)CCCCC1(F)F 25221,c1(C(=O)NCC#CCNC(c2c(C(C)C)n(C)nc2)=O)cc(Cl)c(Cl)cc1O 25222,C(c1ccccc1)=CCNC(COC(CNC(C(C=C)O)=O)(C)C)=O 25223,C(c1cc(C)cc(C)c1)=CC(=O)NCC(CC)NC(=O)CNS(=O)(=O)C1CC1 25224,C1(NC(c2n(CC)ncc2)=O)CC2CCC1N(C(=O)COCc1ccccc1)C2 25225,C1(NCc2cn(C)nc2Cl)CC(O)C12CC(F)(F)C2 25226,Cc1ncccc1C(=O)NCC(C)(C)C(=O)NCC1(n2nccn2)CC1 25227,Cc1c(F)ccc(C(=O)N(C2CCCC(NC(c3c(C)n[nH]c3C)=O)C2)C)c1Cl 25228,c1(CC(N2CC(NC(CC(CCC)O)=O)C3(C2)CC3)=O)c[nH]c2cccc(Cl)c12 25229,N1(C(c2ccsc2Cl)=O)CCC2C(C1)CN2C(c1cnnc(O)c1)=O 25230,c1(CC)ccc(C(N2CCC(CCNC(c3cn(CC)nn3)=O)C2)=O)c(O)c1 25231,CCC(CC)CCC(=O)N(C1C2CN(C(=O)C(C)CC(N)=O)CC12)C 25232,C(=O)(CN=S(C)(C)=O)N(C(c1cnn(C)c1)C(N1CC(N(CCOC)C)C1)=O)CC 25233,c1(CN2CC3N(C(c4c(OC)cncc4)=O)C3C2)c(C)cc(C)cc1C 25234,c1(COC)cc(C(=O)NC(C)(CNC(=O)Cc2nccn2C)C2CC2)no1 25235,O=C1COc2cccc(S(=O)(=O)NCCc3csc4ccccc34)c2N1 25236,CC1(CNC(=O)CC2(O)CCOC2)CCCC1NC(=O)Cc1cnns1 25237,c1(C(N(C(C)C(N2CC3C(N(C)C)C3C2)=O)C)=O)cc(O)ncc1F 25238,C1(C(=O)NCC(C)CNC(=O)CNC(c2ccco2)=O)(CC)CCCCO1 25239,N1(C(c2cc(F)cc(Br)c2)=O)CC2(CCN(C(c3ccc(C4CC4)cc3)=O)C2)C1 25240,C1(CC(=O)NCCNC(C)=O)CCCN1C(=O)CCCN1CCOCC1 25241,N1(C(=O)Cn2cc(C3CCCC3)nn2)CCC2(CCC2)CC1C(=O)O 25242,C#Cc1cccc(NC(=O)CC(C)CNC(=O)CCOCCC)c1 25243,C1(NC(CN2C(=O)CN(C)C2=O)=O)CCC2(CC1)CC2Nc1ncncc1Cl 25244,C(=O)(C(CC(C)C)C(N)=O)NCCCNC(c1ccc(CC)cc1F)=O 25245,c1(CC(C)C)cc(OC(C)C)n(C)n1.c12cc(ncn1)OC1(CCC1)CC(=O)N2 25246,C1(CS(=O)(=O)Nc2cnc(F)nc2)CCCCN1CCc1ccc(Br)cc1 25247,N1(C(C2CC(CNC(=O)C=CCn3cncn3)OC2)=O)CCC(O)CC1C1CC1 25248,C1(NC(N(CC(c2cnn(C)c2)O)C)=O)CC2(C1)CC2NC(=O)OC(C)(C)C 25249,CC1(C)CCCC(O)(C(=O)NC2CN(C(c3nscc3Br)=O)CC2O)C1 25250,C(C)(CCCNC(c1cc(CCO)on1)=O)NC(C1C(C(=O)OC)C=C1)=O 25251,N1(CC(=O)NC(C(C)C)CCN(C(=O)C(F)=CCCF)C)CCCCS1(=O)=O 25252,CC1CCN(C(=O)NC2CCCC2(C)O)C1c1cn(-c2cccc(CO)c2)nn1 25253,C1(O)(CNC(c2c(C)snn2)=O)CCN(C(c2cccc(Cl)c2)=O)CC1 25254,C(N=c1nc2sccc2c(NC2CC(C)CC(C)(C)C2)[nH]1)c1cc(C)cc(C)c1 25255,CCC(CC)C(C)C(=O)N1CC(CNC(=O)CCc2ccc(N)c(F)c2)C(C)C1 25256,C1(C(=O)NCCOC2CCN(C(=O)C(F)n3ccnc3)C2)CC2(C1)CC21CC1 25257,N(C1CCCn2ccnc21)c1cc(NCC2(N(C)C)CCSC2)ncn1 25258,N1(C(=O)NC2CC3(CCCCC3)C2)CC2(CCCC2)c2cccc(F)c21 25259,C1(C(=O)NCC(CN(C)C(c2ccnn2CC#N)=O)O)CCC(C)CC1 25260,C#Cc1cnn(C)c1C(N1CC(C)(NC(=O)CC2CC(O)C2(C)C)C1)=O 25261,n1(C(C(=O)NC2CCC(F)(CNC(C(C)=CC)=O)C2)C)cnc2ccccc12 25262,C(C)(CN=c1nn[nH]n1Cc1ccccc1)NC(C(F)(F)C1(OC)CCC1)=O 25263,C12(C(=O)NC(CCCC=C)C)CC(CN(C(c3ncc(CC)cn3)=O)C1)C2 25264,C1(C(=O)NCCNC(CN(CCC)C(C)=O)=O)CC12CCC2 25265,c12scnc1C1=CCN(CC1)NC2.c1(OC(C)C)ccc(-c2ccccc2)cn1 25266,N1(C(c2cnc(CC)s2)=O)C2CCC1CC(N(C)C(c1cc(C)ncc1C)=O)C2 25267,CCC(CNC(C1CC2(CC2)CO1)=O)(CC)NC(C1CC2CCC2C1)=O 25268,N1(C(CCNC(=O)OC)=O)CC2(CCC(NC(=O)C(C)C(O)CC(C)C)CC2)C1 25269,Cc1nn(C)c(N)c1C(N1CCC(OCC(=O)NC(C)C(O)C(C)C)C1)=O 25270,C(=O)(CC(C)(C)C(C)=O)N1C(C(=O)NC(c2cncc(F)c2)C)(CC)CCC1 25271,c1(C(=O)NC(C(C)(C)NC(C=C(C)Cl)=O)C)ccc(C2(CO)CC2(F)F)cc1 25272,CCCC(CC(C)C)C(=O)N1C(C(=O)NCCC(=O)OC(C)C)C2CC(O)C1C2 25273,C1(C(C)NC(c2cnc[nH]2)=O)CN(C(=O)C(N)=O)CC1O 25274,N1(CC)CC(NC(C2(F)CCN(C(c3nc(Cl)cs3)=O)C2)=O)CCC1=O 25275,CCCCC(O)C(=O)NC1(CCNC(c2[nH]ccc2C2CC2)=O)CCCC1 25276,Cn1cc(C(=O)NCC(C2CCC2)NC(=O)CCC(N)=O)c(-c2ccccn2)n1 25277,S(=O)(=O)(c1c[nH]ccc1=NC1COCC(C)(C)C1)N(CC(CC)C)CC 25278,C1(NC(c2n(CC=C)nnn2)c2cc(C)on2)CCn2nnnc2C1 25279,C1(C(=O)NCCN(C(C23CCC(C2)C3(C)C)=O)CC)CCCC2(CCCCC2)C1 25280,c1(C(N2CCC(NC(COCC#C)=O)C(O)C2)=O)cc(C)c2[nH]nnc2c1 25281,CC1CC(C(=O)NCCC2CC(NC(=O)C3=CCCCO3)C2)CC(C)C1 25282,C1(=CCNC(=O)CC2CCOCC2)CCN(C(=O)CCOCC(F)F)CC1 25283,c1(C(C)(C)C)[nH]cnc1C(=O)NCC(C1CC1)NC(c1cn(CC(F)F)cn1)=O 25284,CC(C)C(C)(CNC(C1SCCS1)=O)NC(=O)Cc1csc(-c2ccoc2)n1 25285,c1(C(=O)NC2C(NC(C(C)NC(=O)NC)=O)C2)c[nH]cc1-c1ccc(C)s1 25286,C1(NC(C2CC23CCC3)=O)CCC(O)CN(C(c2ccc(-c3csnn3)cc2)=O)C1 25287,N1(C(c2c(C)c[nH]c2)=O)CC2CCCC(C1)N2Cc1cc(Cl)ccc1F 25288,C1(N(C(c2cc(C)oc2)C(=O)N(C)C)CCO)CCCN(CCC2CCCO2)C1C 25289,CC(C)CC(O)CC(=O)NC1CCC(C)(CNC(=O)Cc2ccnn2C)C1 25290,c1(C(N)=O)cccc(CC(=O)NCCCCN(CC(=O)NC)CCc2cscn2)c1 25291,c1(C(N(CCNC(c2ccc(Br)o2)=O)CC)=O)ccncc1Br 25292,C1(C(=O)NC(CNC(=O)CCCn2ccnc2)C(C)C)(CSC)CCN(C)CC1 25293,c1(CCC)cc(C(=O)NC2CN(C(=O)CCC(=O)OCC)CC2C)ccn1 25294,C1(CC(=O)NCC2C(NC(CN(C)CCO)=O)CCC2)CCC(F)(F)CC1 25295,N1(C(C2(c3cccnc3)C(C)C2)=O)CCC(COC(=O)C(F)(F)F)CC1 25296,C1(C2CC2)(C(=O)NCC(C(C)C)OC)CN(C(=O)C=Cc2cn(C)nn2)C1 25297,Cn1ncnc1CCC(=O)N(n1ccnc1)CCc1ocnc1C(F)(F)F 25298,c1(CCC)c(C(N2CCC(CF)(NC(c3nocc3C)=O)C2)=O)cnn1CCO 25299,c1(C(N(CC2CCN(C(C34CC(CCC)(C3)C4)=O)C2)CC)=O)cn(C)[nH]c1=N 25300,C1(NC(c2ccn(C)c2)=O)CC(NC(c2nnc(S)n2C)=O)C12CCC2 25301,N1(CC)CC2CC1CN2C(C1(CNC(c2cscc2Cl)=O)CCCC1)=O 25302,C1(NC(CC(C)c2ccco2)=O)COC2(C1)CN(C(=O)CC1CC(F)C1)C2 25303,C(C)(CNC(=O)C(O)CC1CC1)(CC(C)C)NC(c1[nH]cc(C)c1)=O 25304,Cn1ccc2cccc(C(=O)NC3(C)CCN(C(c4sccc4F)=O)C3)c12 25305,C(CCN(C)C(c1ccn(C2CC2)n1)=O)(C(C)(C)C)NC(c1c(C)cno1)=O 25306,C(=O)(CCCCCCNCc1occ(C(=O)Nc2c(C)ncnc2)n1)OCC 25307,CCCCC(C)CCC(=O)NC(COCC)C(=O)N(C1CC=CC1)C 25308,N1(C(C2N(CC)CCC2)=O)CC(C)(C)C(NC(C2CCOCC2)=O)C(C)(C)C1 25309,N1(C(=O)NC2(OC)CC(OC)C2)CCC2(CC1)CC2NC(=O)OC(C)(C)C 25310,c1(NC(CC2CCCN(C(C(CC=C)C)=O)C2)=O)ccc(Cl)nc1C(N)=O 25311,c1(C(N(CCNC(C=C(CC)C)=O)CCOC)=O)cccc(F)c1Br 25312,C12(C(=O)OC)CCN1C2=O.C1(OC)CC(C)N1C(=O)OC(C)(C)C 25313,CCC(O)C(F)(F)C(=O)NCC(C1CCN(C(c2ccncc2F)=O)CC1)C 25314,C1(CC)C(C(=O)NC2CCN(C(=O)CCCn3nc(C)nc3C)C2C)CCN1C 25315,C12(CC(N3CCC4CN(C(CC=C)=O)CC4C3)=O)CC3CC(C)(C1)CC(C)(C3)C2 25316,C(=O)(C(C)C(O)C(C)C)N(CC(COC)C)C.C(=O)C(C)(C)C1CCCC1 25317,N1(CC(C2CCOCC2)CC)CCC(c2nc(C(=O)OC)n[nH]2)CC1 25318,c1(C(=O)NCC(C)CNC(C2(F)CCOC2)=O)nc(Br)c2c(F)cccn12 25319,N1(C(CCc2ccc(C)o2)=O)CCCC2CN(C(=O)C(C)(C)C(C)(C)O)CCC12 25320,S(=O)(=O)(c1cccc(Cl)c1F)NC1CCC(C(=O)NCc2ccc(O)cc2)OC1 25321,c1(C(CO)NC2CC(C)(CC)C2)ccc(F)cc1F 25322,N1(c2n(C)nnn2)CCC(NC(=NCc2ccn(C(F)F)n2)NCCF)CC1 25323,C(CC(=O)NCC(C)CN(C(=O)CCc1ncco1)C)OCCC 25324,C1(F)(CNC(=O)Cc2c[nH]nc2O)CCCN(C(C2(CC3CC3)CCCO2)=O)C1 25325,c1(C(N2C3CN(C(C4(C=C)CC4)=O)C(C3)C2)=O)cc2ccc(OC)cc2s1 25326,C(CCCCC(=O)NCC1CCCC(C)(C)C1)N(C(=O)C1=CCCCC1)C 25327,CC1(C)CN(C(c2cc[nH]c(=N)c2)=O)C(CNC(C2CCCN2C2CC2)=O)CO1 25328,C(=O)(C1=C(C#N)CCC1)NC(C1CCCN(C(c2c(C)nc(N(C)C)s2)=O)C1)C 25329,c1(C(N2C3C(NC(=O)CCC4CCCO4)C(C3)C2)=O)n[nH]c2c1CCC2 25330,C1(NC(C(C)OCC(C)C)=O)CC2CC(C1)CN(C(C1(O)CC(C)(C)C1)=O)C2 25331,O=C1CC2CN(C(C3CCCN(C(=O)Cn4ccnn4)C3)=O)CC2CN1 25332,C=C(F)C1(CC(=O)NC2CCCCC2N(C(=O)C(C)SCCCC#N)C)CCC1 25333,n1(CC)cc(Br)cc1C(=O)OCc1nnc(C2CC2)o1 25334,Cn1cc(Cl)c(C(N2CC(O)(CCNC(C34COCC3C4)=O)C2)=O)n1 25335,C1(CC)CCN(C(c2[nH]ccc2CNC(=O)CCCCSC)=O)C1C 25336,c1(C(N2CCC2)=O)cc(S(=O)(=O)NC2CC3(C2)CC(Br)C3)c[nH]1 25337,C1(C(C)O)CCC(NC(C2CCC(C(=O)O)N2C(c2ccc(Cl)cn2)=O)=O)CC1 25338,N1(C(c2c(C)nsc2)=O)CCC(C)C(NC(C2(F)CCCCC2)=O)C1C 25339,N(C(=NCCc1cnccc1OC)NC1COC(C)C1)CCC(=O)NC 25340,c1(C(=O)NC2C=CCN(C(C3(C)ON=C(C)C3)=O)C2)cccc2ccnn12 25341,C#Cc1c[nH]nc1C(=O)NC(C)CC(C)NC(=O)Cc1ccc(F)cc1 25342,C1(NC(C(COC)NC(C)=O)=O)CC2(C1)CC(NC(=O)CSC(F)F)C2 25343,C1(NC(C(c2cncnc2)C)=O)(CO)CCCN(C(c2cc(Cl)no2)=O)C1 25344,Cc1nc(N(C)C)sc1C(=O)NC1CCC(CCNC(C2(O)CCSC2)=O)C1 25345,C=Cc1cnn(C)c1C(=O)NCc1cccc(NC(C2(C)CCC(C)C2)=O)c1 25346,C1(NC(C(C)OC(C)=O)=O)CC(CC(=O)NC2(CC(C)(C)C)CC2)C1(C)C 25347,C1(C(N2C(C3(NC(COCCC)=O)CC3)CCC2)=O)CC(=O)N(CC(F)(F)F)C1 25348,CCCCCC(O)CC(=O)N1CCOC(CNC(=O)CC2CC=CCC2)C1 25349,c1(CN2CCC(N(CCOC)C=O)C2)cccc(OCC2CCOC2)c1.C1CC1 25350,C(=O)(C(Cn1cccn1)NC(=O)CC1CCCC1)NCC(C)OC 25351,C1(NC(c2ccc(OC)o2)=O)CC2CC1CN(C(=O)Cc1ccc(F)cn1)C2 25352,c1(NC(C2CC2Cc2cccnc2)=O)cnn(Cc2ccccc2)c1 25353,c1(CC)nc(C(N2CCC(CCNC(C34CC(O)C3C4)=O)C2)=O)co1 25354,N1(C(C2N(CC)CCC2)=O)CCCC(CNC(=O)CN2CC(C)(OC)C2)C1 25355,Cc1ccc(C(N2CC(O)(CCNC(C3CN(C)C(=O)CCO3)=O)C2)=O)cc1C 25356,c1(N2CC(F)(C(=O)Nc3cc(COC)ncc3)C2)ncnc2cnccc12 25357,c1(C(=O)NC(CCNC(C(C)SC(C)C)=O)C)ccc2c(c1)NC(=O)CN2C 25358,N1(C(C(CNC(c2cnn(C)c2Cl)=O)CC2CC2)=O)CCC(O)(CO)CC1 25359,c1(Nc2c(C)cc(N3CCSCC3)cc2)nc(S(C)(=O)=O)nc2c1ncn2C 25360,N1(C(COC)=O)CC(NC(c2nc3cccnc3s2)=O)CC12CCCOC2 25361,c1(C(=O)NCc2c(C(N3C(C)(CCC)CC3)=O)occ2)nc(C)ccc1C 25362,C1(CNC(CC(CCOC)(C)C)=O)CCC2CN(C(=O)C3=CCCO3)CCC2C1 25363,C(=O)(C(CNC(=O)Cc1cncn1C)N(C)C)NCC(N(C)C)C1CC1 25364,S(=O)(=O)(c1ccc(NC(c2cccs2)CC)nc1)NC(c1ccc(Cl)cc1)CC 25365,c1(C(=O)NC(CNC(c2c(SC)cc(F)cc2)=O)(C)C)cc2ccc(F)cc2o1 25366,C(=O)(C1OCCc2cc(Br)ccc21)NCCNC(c1c(OC)scc1)=O 25367,c1(OC)c(NC(c2cnn(CCN(C)C)c2)=O)cccc1SC 25368,C1(NC(CCc2nc(C)sc2)=O)COC2(C1)CN(C(C1CC1C1CCCC1)=O)C2 25369,C(=O)(C1CCCc2nncn21)N1C(CNC(C2CC2(Cl)Cl)=O)CC2(CC2)C1 25370,C12C(C3CC3)CCN1C(=O)CC(C)CC(=O)NC2.C(C(O)C=O)=CCCC.OCC 25371,Cc1ccc2c(c1)C(C(=O)NC(C)CNC(c1ccc(CO)cc1F)=O)C2 25372,CC1(C(N2CCC(C)(NC(c3cc(F)cnc3O)=O)C2)=O)CCCCC1(F)F 25373,Cc1cccc2[nH]cc(C(=O)NCC3CC3NC(c3nnc(O)nc3O)=O)c12 25374,C1(NC(c2[nH]cc(CC)n2)=O)CCC2(CCN(C(=O)CC(C)CC(C)(C)C)C2)C1 25375,c1(C(C)N)ccc(N(CC(=O)OCCCC#N)C(=O)CC)cc1 25376,Cc1cc(C(N2CCC(N(CCO)C(c3cn[nH]c3)=O)C2)=O)n2ncnc2n1 25377,c1(-c2ccc(C(N3C(CCCNC(C=C(C)C)=O)CCC3)=O)s2)cccc(F)c1 25378,Cc1cccc(OCC(=O)NC(CNC(=O)C2=CCCSC2)CO)c1C 25379,C1(O)(CCNC(c2n[nH]cc2F)=O)CCCN(C(c2sccc2C(F)F)=O)C1 25380,C1(NC(C(CC=C)OC)=O)CC(NC(C23COCC(C2)C3)=O)C12CCC2 25381,C1(Cn2cnc(CC)n2)CCN(C(=O)Cn2cc(I)nn2)CC1.c12cn(nn1)C2 25382,c1(CNC(C(CC)(C)C)=O)cc2n(n1)CCN(C(=O)CN1CCCNS1(=O)=O)C2 25383,C1(F)(CNC(=O)C(F)=CC2CC2)COCCN(C(c2ncsc2C2CC2)=O)C1 25384,n1(CCNC(=O)NCC2(C)C(C)(C)C2)ccn2nccc2c1=O 25385,O(NC(=O)C(CC(N)=O)NC(c1csc(C#N)c1)=O)CC(=C)Cl 25386,C1(C)(CC)NC(=O)N(CC(N2CC(F)CC2CNC(=O)C(C)(C)C2CC2)=O)C1=O 25387,c1(CC(=O)NC(CNC(C(CC)F)=O)(C)CO)cccc(NS(C)(=O)=O)c1 25388,c1(-n2cc(CNC(c3ccc(C(CC)C)cc3)=O)nn2)cc(C)c(F)cc1Cl 25389,N1(C(c2ccc(C(C)C)s2)=O)CCC12CN(C(=O)CC13CCCC1C3)C2 25390,CC1(CNC(=O)CCC2(NC(=O)C=CC(=O)N(C)C)CCCC2)CCCCC1O 25391,c1(C(=O)O)ccn(CC(N2CC(c3cn(CCCCCO)nn3)C2)=O)n1 25392,N1(C(=O)NCCN2CC(C)C2)CCC(C)C1c1ccc(C(F)(F)F)cc1 25393,C1(C(N2CC(OCCNC(CCOCCNC(C)=O)=O)C2)=O)(CO)CCCCO1 25394,C1(CNC(C2C(C)=C2)=O)C2CN(C(=O)COc3ccccc3)CC12 25395,C(CN=C(NCC1(O)CCN(C)C1)N1CCC(CSC)C1)CCC=C 25396,C#CC1CN(C(=O)CC2CCC(C)(C)O2)CCN1C(c1nnsc1SC)=O 25397,N1(CC)CCC(CNC(=O)CC2C=CC(NC(=O)C=C3CCOCC3)C2)CC1 25398,N1(C(CCSCC)=O)CCOC2(CCN(C(=O)CN3C(=O)CNC3=O)C2)C1 25399,c1(SC)nc(N2CCN(C(=O)C(N3CCCC(C)C3)=O)CC2)ncc1F 25400,C(C(CC(=O)N1CCC1c1cccnc1)C1CCC1)NC(=O)C(C1(O)CCCC1)F 25401,C1(CNC(c2c(C)nn[nH]2)=O)CC(F)CN1C(c1cc(I)on1)=O 25402,C1(O)(CNC(c2c(C(C)C)cco2)=O)CCCN(C(=O)CCC2CCC(=O)N2)C1 25403,N1(C(c2c(C)nccn2)=O)CCC(C2CCCN(C(=O)C(C)(F)F)CCC2)CC1 25404,c1(C(=O)NC2CC(CCNC(CC(COC)C)=O)C2)cnn2ccccc12 25405,C(=O)(CC1=CCOCC1)NC(COC)C(=O)NCC1CCC(C)CC1 25406,c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)C2)ccc(C(C)C)cc1F 25407,CC1(CC(=O)NCc2ccccc2Cl)CCN(C(C2(C)CCCC2O)=O)C1 25408,c1(NCC2(O)CCCN(C(C(CC)OC)=O)C2)c(C#N)cnc2c(Cl)cccc12 25409,Cc1cc(C(=O)N(C2CC(NC(=O)C(C)NS(C)(=O)=O)C2)C)sn1 25410,C(=O)(CCCCC(C)(C)C)NC(C(C(C)C)NC(=O)C=Cc1ccc(F)cc1)C 25411,N1(C(c2ccc(C)nc2C2CC2)=O)CC(C)N(C(=O)CN(C)C2CC2)CC1C 25412,CC(C(=O)NCC1CCOCC1)C(C)NC(C1C2CC(=O)CC12)=O 25413,C1(C(N2C(c3cn(CC4CCC(=O)O4)nn3)CCC2)=O)CC2CCCC2C1 25414,CC(CC(C)NC(=O)CCCF)NC(=O)C(CC1CC1)NC(=O)OC(C)(C)C 25415,C1(COC)CCCCN1C(=O)CCN(C(=O)CCc1ccc[nH]1)C(C)C 25416,CC(C)(F)CCC(=O)NCC1(C)CCCN1C(C1COC(=O)O1)=O 25417,CCCCS(=O)(=O)CC(=O)NCC1CCN1C(c1ccn2ncccc12)=O 25418,C1(C(=O)NCC(COC)NC(c2cnc(C3CC3)s2)=O)CNC(=O)N1C 25419,C=CCC(C)(C(F)F)NC(=O)CCn1cc(-c2ccc(C)cc2C)nn1 25420,C1(NC(c2ccn(CCOC)n2)=O)CN(C(=O)CNS(=O)(=O)C2CC2)CC1C 25421,S(=O)(=O)(c1ccc(OC)cc1O)NC1CCC(NCc2ccc(OCC)nc2)C1 25422,Cc1cc2[nH]c(C(=O)NCC(C(C)C)NC(=O)CCCCCN(C)C)cc2o1 25423,c1(C(=O)NCC(C2CCCC2)C)cn(CCNC(c2cc[nH]n2)=O)cn1 25424,N1(C(CCNC(=O)CO)=O)CCC(C2CCN(C(c3ncc(Cl)cc3F)=O)C2)C1 25425,N1(C(c2n(CCC)ccc2)=O)CC(CNC(C2(C)CCCCC2)=O)CC12CCC2 25426,N1(C(=O)NC2CCC(C)CC2)CCN(CC(C)NC(CC=CCC)=O)CC1 25427,n1(CC(=O)NCCCN(C(=O)C(O)CC[S+](C)C)C)c(O)nc2ccccc12 25428,c1(C(=O)NC(CC(C)NC(CC(CC)(F)F)=O)C)cc(S(N)(=O)=O)c[nH]1 25429,c1(CN(C(=O)NC(c2cccc(F)n2)C)C)cccc(Cl)c1Cl 25430,Cc1cc(C)c(C(=O)NCCC2CCN(C(=O)C(c3ccccc3)O)C2)s1 25431,C1(C(=O)NCC(CNC(C2(N(C)C)CCC2)=O)F)C2CCC3(COC(=O)C13)O2 25432,Cc1cnc(C(N2CCC(C)C(NC(c3cccnc3O)=O)C2)=O)c(F)c1 25433,C(=O)(C(C(C)O)NC(C)=O)NC(CC)CNC(=O)C(C)c1ccon1 25434,C12(CC)CCN(C1)c1nnc(C3CC4C=CC3C4)n12.N12C(CCC1C)C2=O.CSC 25435,C1(C(N2CCC(N(C(=O)CCCCc3ccccc3)C)C2)=O)CCC(C)(F)CC1 25436,Cc1nsc(C(N2CCCCC2CCC(=O)N(CC(C)C#N)C)=O)c1N 25437,N1(C(c2c(OC)n[nH]c2)=O)C2CCC(C2)C1CNC(C1CCC(C)(C)CO1)=O 25438,Cc1nc(NCC(C)(C)C)cc(=NCc2ccc3ncsc3c2)[nH]1 25439,c1(C(=O)NCC(C)NC(C(CC)OC2CCCC2)=O)c(C)oc(C)c1S(N)(=O)=O 25440,C(CNC(c1cnc(SC)s1)=O)(C(C)(C)C)NC(c1cn(CC(CC)O)nn1)=O 25441,Cc1cc(F)cnc1C(=O)NC(C1(C(=O)NCC2CC(C)(C)C2)CC1)C 25442,C1(C(=O)NC2C(NC(c3nc(C)oc3)=O)CCCC2)CCCC2(CCC2)O1 25443,N1(C(c2c(CNC(C(C)SC(C)C)=O)nccc2)=O)CCc2nnnn2CC1 25444,C1(O)(CNC(C2CCN(C(CC)=O)C2)=O)CCN(C(c2cnoc2CC)=O)CC1 25445,c1(C(=O)NC2C(C)(CNC(C3(O)CCOCC3)=O)CCC2)nnc(O)cc1O 25446,C1(C(N(CC(CN(C(COCC(C)C)=O)C)O)C)=O)Cc2ccccc2S1(=O)=O 25447,c1(C(=O)NC23CC(CNC(c4c(CC)occ4C)=O)(C2)C3)ccc2c(c1)CCO2 25448,N1(C(CCCCC=C)=O)CC2CC1CCC2NC(c1csnc1Br)=O 25449,C(=O)(CCCC(C)(c1nnnn1C(C)(C)C)NC1(C)CC=CCC1)OC 25450,C1(N(C(CCCOC)=O)C)CC2CCC(C1)N2C(C12CCCC1C2(F)F)=O 25451,C(CC1CCCO1)(CC)NC.C12(F)CC1CN(C(C=CCCC)=O)C2=O 25452,N1(C(c2cc(CNC(c3ccco3)=O)no2)=O)CC2CC1C(F)(F)C2 25453,N1(C(C(CC(=C)C)C)=O)CCC2CCN(C(c3c[nH]c4nccc-4c3)=O)C2C1 25454,C1(C(N(CCCNC(c2c(C)oc(Cl)n2)=O)C(C)C)=O)CCOC(=O)CC1 25455,C(=O)(C1=C(CC)OCCS1)NCC(C1CC1)NC(c1oc(CC)c(C)c1)=O 25456,C(=O)(CC1COc2ccccc21)NC(C)CN(C(=O)Cn1cc(C(F)F)cn1)C 25457,C(C(C)CC(=O)N1CCCCC1C(C)(C)CNC(c1cc(C#N)on1)=O)OC 25458,N1(C(C2(CNC(c3ccc(C)o3)=O)CCCO2)=O)CCCC(C)CC1 25459,c1(CNC(c2c(C)cns2)=O)cncc(C(=O)N(C2CCCCC2C)C2CC2)c1 25460,C1(OC)CCC2(C(N3CCCC(CNC(c4cnn(C5CCC5)c4)=O)C3)=O)CC12 25461,c1(CCC)cc(C(=O)NCC(O)CCNC(=O)Cc2cccn2C)ccn1 25462,CC1c2cc(O)ccc2CCN1C(=O)Nc1snc(-c2ccccc2)c1Cl 25463,c1(C(=O)NCC2C3CN(C(C4(CCCC)CC4)=O)CC32)cc(CC)nnc1C 25464,c1(CCC(=O)NC2CN(C(CCC(=C)Cl)=O)CC(C)C2)cccc(S(N)(=O)=O)c1 25465,C1(CNC(CN(C)CCO)=O)CN(C(C2CC3CCCC3C2)=O)CC(C)(C)O1 25466,C1(C(C)(C)NC(=O)CN2CCCC2=O)CCN(C(C2COC(=O)O2)=O)CC1 25467,c1(CC)cccc(C(=O)N(CCCN(C)C(c2ccc(O)nc2)=O)C)c1O 25468,Cc1cc(C(=O)NC2CC(C(N3CCC(CCF)CC3)=O)C2)ncn1 25469,N1(C(C(C)OC)=O)CCC2(CC1)CC(N=c1[nH]c3cc(F)ccc3o1)CO2 25470,N1(C(CCCOCCOC)=O)CC2CN(C(C34CCC(C3)OC4C)=O)CC(C1)O2 25471,CS(=O)(=O)C(CNC(=O)CCSCC(N)=O)CNC(C1CC2CCC2C1)=O 25472,C12(CC(=O)NC3CCN(C(c4ccc(CO)cc4)=O)C3)COCC(C1)C2 25473,N1(C(c2nc(CC)oc2)=O)CCC(C(=O)NCC2CCC(=O)NC2C)CC1C 25474,N#Cc1c(NC(=O)CCC(=O)C(O)CC2CCNCC2)sc2c1CCC2 25475,c1(OC)ccc(CCNC(C23CC(C(=O)NC(C)(C)C)(C2)C(C)O3)=O)cc1OC 25476,C(=O)(C1SCCc2sccc21)OC(C(C)(CN(C)C)NCCC#N)C 25477,C12(NC(c3cnc(=N)[nH]c3)=O)CCN(C(c3cnn(C4CCCC4)c3)=O)CC1C2 25478,CN1CCCC1CCC(=O)N1CC(OCCNC(C2CCN(CC(F)(F)F)C2)=O)C1 25479,C(=O)(C1CCCc2nn[nH]c21)N1CC2CC(NC(=O)Cn3ncccc3=O)C2C1 25480,Cc1cc(-c2nc(C)c(C(=O)NS(=O)(=O)c3cccc(Br)n3)s2)cc(C)c1C#N 25481,c1(C(N2C(CNC(c3c(C)ccc(OC)c3)=O)CC2)=O)cn(C)c2ncccc12 25482,CCCCCC(O)C(=O)NCC(O)CNC(=O)Cc1ccc(CCCC)cc1 25483,N1(C(c2cc(C)no2)=O)CC(C)CN(C(c2cc(C(F)F)nn2C)=O)C(C)C1 25484,C1(CC(=O)NC(C)(C)CF)(OC)CN(C(C2CC(=C3CCC3)C2)=O)C1 25485,c1(CC)c(C(=O)NC2COCCC2C(=O)NC(c2cccnc2)CO)ccn1C 25486,c1(C(=O)NCC2C(NC(c3c(C)snc3)=O)COC2)nc(C2CC2)oc1C 25487,Cn1c(NCC2(CNC(=O)CC=C(Cl)Cl)CCC2)cc(=O)n(C)c1=O 25488,c1(CNC(CN(C(C2(O)CCSC2)=O)CC)=O)cc(CO)[nH]n1 25489,N1(C(C2(S(C)(=O)=O)CCC2)=O)CC2CCC1CN2C(=O)CN1CC2C=CC1C2 25490,CC1CCCC1NC(=O)CCCN(C(=O)CC1CCCC1)C 25491,c1(CNC(c2cc(C)[nH]n2)C)ccc(CN2CCN(C)CC2)cc1 25492,N1(C(c2n(C)nc(Br)c2)=O)CCC(NC(=O)CCc2cnco2)C12CC2 25493,C1(SC)CC(CC(=O)NC(C)CCN(C(=O)C(C)C)C)C1 25494,N1(C(C(C)OCC=C)=O)CC(OC)C(CCn2cc(-c3ccc(C)cc3)nn2)C1 25495,c1(C(=O)NCC(CO)NC(CC(CC)C2CC2)=O)cc(C)ncc1C 25496,N1(C(CC=C)=O)CCC2CCCC12C(=O)NC(c1ccnn1C)C 25497,S(=O)(=O)(c1ccc(C(=O)NC2CC(NC(C3CC3(F)F)=O)C2)cc1)N(CC)CC 25498,CS(=O)C1CN(C(=O)CC2CCN2C(c2csc(Cl)n2)=O)C1 25499,c1(C(=O)NCCCC2(CNC(C(C)N(C)C)=O)CCCC2)cnc2ccoc2c1 25500,CC1CNC(C)(C)CN1C(=O)Cc1ncc(Br)s1 25501,C=CC1(C(=O)NC2CCC(NC(=O)C(C)=CCC)CC2)CCCCC1 25502,C(=O)(CCCN=[N+]=[N-])N1CCC(N(C)Cc2c(C(=O)OC(C)(C)C)occ2)CC1 25503,CN1CCN(C(=O)CC2CCCC(C)(C)C2)CC1CNC(c1ccnnc1O)=O 25504,C1(CNC(CCc2n(C)ccc2)=O)C(O)C(O)CN1C(C1CCNC(=O)C1)=O 25505,c1(C(=O)NCC2C(NC(=O)CNC(N3CCCC3)=O)C2)cnc2ncccc2c1 25506,N1(C(CSCCCC)=O)CCC(C)(CNC(=O)C2=NOC(C(C)(C)C)C2)CC1 25507,C(=O)(CC(CC(C)C)NC(C12CCC(C)(C1)OC2)=O)N1CC(C)(CC=C)C1 25508,N1(C(C)C)C(=O)CCC1C(=O)NCCCNC(=O)CC1CC2(COC2)C1 25509,C1(C)(C(=O)NC2CC(C)(OC)C2(C)C)Cc2ccc(Br)cc2C(=O)O1 25510,Cc1ncncc1NC(C1CC1NCc1cccc(CO)c1)=O 25511,N1(C(c2n(C)ccn2)C(=O)NC2CC(F)(F)C2)CCC12CC(C(N)=O)C2 25512,C1(C(=O)NCC2(NC(C3CC34CCCC4)=O)CC2)(CC)CNC(=O)C1 25513,Cc1cc(CCC(=O)N(CCNC(=O)CC2(C)CC2(F)F)C(C)C)on1 25514,C1(NC(C(C(C)C)(C)C)=O)CC2CCC1CN(C(=O)CC1CCCCC1O)C2 25515,c1(C(=O)NCCN(C(CCn2ncc(C)c2)=O)CC(C)O)cc2ccncc2s1 25516,N1(C(c2c(C)cn(C)c2)=O)CCC(F)C(NC(c2cc(C)n(C(C)(C)C)n2)=O)C1 25517,c12cc(sc1C)C(=O)NCCN(CC(C)O)C(=O)CNC2=O.C1(CC)CCSC1 25518,Cc1nn(C)c(C)c1CCC(=O)NCCOCCCNC(=O)CC1CCCOC1 25519,c1(OCC)cc(CNC(=O)NC2(c3cc(Br)nc(Br)c3)CC2)ccc1OC 25520,N1(C(c2c(C)csc2)=O)C2CCCC1CN(C(C1CCc3n[nH]cc3C1)=O)CC2 25521,C1(C(N2C(C(C)C)C(C)(C)C2)=O)CN(C(C2CC(C)(C)CO2)=O)CC1(F)F 25522,N1(C(C(c2ccc(C)cc2)C)=O)CC2(C1)CN(C(=O)C(C)(C)CF)CCO2 25523,C1(C(N2C3C(NC(CN(CCC)C)=O)C(C3)C2)=O)CCCC2CCCN12 25524,c1(C(=O)NCCN(C(C(CC#C)O)=O)C2CC2)ccc(OC)c(C)c1 25525,c1(C(=O)NC2CC23CCN(Cc2cncc(Br)c2)CC3)ccc(I)c([N+](=O)[O-])c1 25526,N1(CC)CCN(C2CCCN(C(=O)C(C(C)C)NC)C2)C(=O)C1.OC 25527,c1(C(N(C)CC2N(C(CS(=O)(=O)NC)=O)CCC2)=O)cc(N)cnc1Cl 25528,C1(C(N2CC(S(C)(=N)=O)C2)=O)(NC(c2scc(OC)c2)=O)CCC(C)(C)C1 25529,c1(N2CC(N(C(c3ccn(CCOC)n3)=O)C)C2)ncnc2[nH]c(C)nc12 25530,c1(C(=O)NCC2CC(NC(C(C=CC)O)=O)C2)cc2n(n1)CCCC2O 25531,Cc1ncc(Cl)cc1NC(=O)COC(C1CC1c1ccc(C2CCCCC2)o1)=O 25532,c1(-c2nc(C(=O)Nc3nc(NC(C)=O)nc(O)c3)sc2)ccc(Cl)c(C)c1F 25533,C(=O)(CC(C)C(C)C)NC(COCC)C(=O)NC1CCC(CC)CC1 25534,C(=O)(CC(C)(C)N(C)C(C1(Cl)CC1(F)F)=O)N1C(CCCC)CCC1 25535,C1(C#N)(C(=O)NCCCCCN(C(c2c(C)n[nH]c2)=O)C)C(C#N)C1(C)C 25536,C1(C(=O)NC2CCCC(NC(c3ccc(C(F)F)nc3)=O)C2)CCCC12CCC2 25537,N1(C(c2c(C(=O)OC)c(C)[nH]n2)=O)CCCC(C2CN(C(C3(SC)CC3)=O)C2)C1 25538,C=CCC(CNC(=O)C(C#N)CCC)C(=O)N1CCC(OC(C)=O)C1 25539,c12cc(ncn1)N(C1CNCC1C#N)C2=O.c1(CC)cc(Cl)sc1Cl 25540,c1(NC(C(C(C)(C)C)N(C)C)=O)ccc2nc(NC(c3ccccn3)=O)sc2c1 25541,C1(CNC(c2ccc(Cl)[nH]2)=O)CC(F)CN1C(C1CCS(=O)(=O)C1)=O 25542,CN1CCC(=CC(=O)NC2CC(CCNC(c3n[nH]cc3Br)=O)C2)CC1 25543,Cc1nc(C(C)NCC2CN(C)CCO2)ccc1OC(C)C 25544,CC1(CNC(c2cc(Cl)ccc2F)=O)CN(C(C2CCOC2=O)=O)CCO1 25545,C=CCCC(C(=O)N1CCOC(C)(C)C1)NC(=O)CCn1cnnn1 25546,c1(C(=O)NCC2CCN(C(C)C)C2)ccc(F)c(F)c1F.c12cc(ncn1)N2 25547,C12(CNC(C)=O)CC1CN(C(=O)NC(CC(C)C)c1nc(CNC(N)=O)no1)C2 25548,N1(C(C2CCC(C)O2)=O)CCC2(CCC2NC(=O)Cc2ccco2)CC1 25549,Cc1cc(NC2CC(F)(CNC(C3(C(F)(F)F)CC3)=O)C2)c(Br)cc1[N+](=O)[O-] 25550,CC(C)(C)CCCC(=O)NCC(C)(C1CC1)NC(C1CC2(C)CC1CO2)=O 25551,C1(C(=O)NC(CCSC)C)CCN(C(=O)CCCC2CCCO2)O1 25552,C1(C(N(C2CC(OCC)C2)C)=O)CCN(C(=O)CC2(CSC)CC2)C1 25553,c1(C(N2CCC(NC(C(CCC)OCC)=O)CC2)=O)c(C)nn(C)c1N 25554,c1(C(N2CC3(CCC(NC(CC=C)=O)C3)C2)=O)cc(C)cc([N+](=O)[O-])c1 25555,C(=O)(C1Cc2c(Cl)cccc21)NC1C(F)CCN(C(c2ccc(SC)s2)=O)C1 25556,c1(N2CCC(CC=C)(NC(C)=O)C2)nc(O)c2cnn(-c3ccccc3)c2n1 25557,C(=O)(C1CCc2c[nH]nc21)N1CCC(CC(=O)Nc2cc(C)nc(O)c2)C1 25558,c1(CC(=O)NC2CN(C(C(CSC)O)=O)C(C)CC2)cccc([N+](=O)[O-])c1 25559,C(=O)(C(C)(CCC(F)(F)F)c1ccccc1)NCc1nc(C)c(C)[nH]1 25560,c1(C(N(CC(C)CNC(c2cnsc2)=O)C)=O)cc2c(nc1O)CCCC2=O 25561,C1(n2ncc(C)c2)CCN(C(=O)C(=O)Nc2cnn(CC3CCCOC3)c2)CC1 25562,c1(OC)cc(CN2CCN(c3nc(N(C)C)cc(C)n3)CC2)ccc1Cl 25563,C1(NC(c2nc[nH]c3nccc2-3)=O)CN(C(=O)C=CC2CCC2)C2CCCCC12 25564,C=CCC(CNC(=O)Cn1cc(C)cn1)C(=O)NCC1(CO)CC12CCC2 25565,C1(N(C(=O)CCc2cnoc2)CC)CCCN(C(=O)CC=C(C)C)C1 25566,c1(COC)nc(NCCc2c[nH]nc2O)cc(=NC2CCCC(C)C2)[nH]1 25567,c1(CC2(SC)CC2)ccccc1.C(C)(CC(C)C)N1CC1=O 25568,C1(NCC)CC(C(=O)OC(C)(C)C)N(C(C2(CNC(=O)CS(C)(=O)=O)CC2)=O)C1 25569,c1(OCC)nc(C(=O)NCC2CN(C(C3(C)CC3)=O)CC2OC)cc(O)n1 25570,N1(CC(=O)N(C(C)C(=O)NCC(F)(F)F)CCC)CCc2sccc2C1 25571,C(CCCCC(=O)NCC(CNC(C1CC(C)(C)O1)=O)OC)OCC 25572,N1(C(C(C)(CO)OC)=O)CC2(C(=O)Nc3cncc(C4CC4)c3)CC1CO2 25573,N1(C(c2cccc(C(F)(F)F)n2)C(=O)NC)CC(N=[N+]=[N-])CCC1(C)C 25574,C=CCCCCCC(=O)N1CCC2(NC(=O)Cn3cc(CN(C)C)nn3)CC2C1 25575,n1(-c2cc(C)on2)c(C)cc(C=CC(=O)NC2CNC(=O)C(C)(C)C2)c1C 25576,CC1CCN(CC(C)(C)COC(C2(c3ccc(SC(F)F)cc3)CC2)=O)CC1 25577,c1(NC(C(CC)C)C)ccc(S(=O)(=O)NCc2cccc(F)n2)c(Br)c1 25578,C1(CNC(COC2(C)CN(C(=O)CC3COCCO3)C2)=O)CCCC(CO)C1 25579,CC1(C)COc2c(C(=O)NCC3CC3NC(c3csc(C#N)c3)=O)cccc21 25580,N1(C(c2c(Cl)ccc(C#C)c2)=O)CC2CCCCC2(NC(C2CCN(C)C2)=O)C1 25581,c1(-n2cc(C(N3CC(NC(C(CC)OC)=O)C(C)C3)=O)nc2)ccc(Cl)c(Cl)c1 25582,C1(CN(C(C2CC2CC(C)C)=O)CC)CCCCN1C(=O)CC1(OC)CCC1 25583,Cc1ccc(OC(C)C)cc1NC(c1cnn(C2CCOCC2)c1C)=O 25584,N1(C(c2c(CCC)cccc2)=O)CC2CCC2(CCNC(=O)C2=CCCCC2)C1 25585,C(=O)(CCCCCC(=O)NC(C)CNC(=O)CC1CCC2(CC1)CC2)OC 25586,C1(OCC)CCN(C(=O)C=CC(C)(C)NC(=O)CCOC(C)=O)CC1C 25587,C12(CCNC(CCc3c(C)noc3)=O)CCC1CN(C(c1cncs1)=O)C2 25588,Cc1cc(CC(N2CCCC2CCNC(=O)Cc2cccnc2C)=O)ccc1O 25589,CCCC(O)CC(=O)NC1CN(C(c2ccnn2CCC(F)(F)F)=O)CC1O 25590,c1(C(=O)NCCc2cn(-c3n(C)nnc3)nn2)cc2cc(Br)cn2cn1 25591,n12cc(c(=O)cc1C)C(=O)NC1CCCCC1CC2.C(=O)(CCS(N)(=O)=O)OC 25592,c1(C(=O)NCCC2CC(NC(c3nn(C)c(O)c3)=O)C2)cnc2ncccn12 25593,C12(NC(C=CC(C)NC(C(CC)=CC)=O)=O)CCN(CC1)CC2 25594,c1(NCC(CCCC)NC(=O)Cn2ccnn2)ccc([N+](=O)[O-])cn1 25595,N1(C(C(C(=O)OCC)OC)=O)CCC2(CCN(C(=O)C=Cc3ccco3)CC2)C1 25596,C12(CCCSC1)CN2.N1(C(=O)NCC)CCCCC1CN 25597,C1(NC(C2CCCN(C)C2)=O)CC2CC(NC(=O)CC3(C)CCOC3)C2C1 25598,C1(C#N)(C(N(C2CC(c3cn(C4(O)CCOCC4)nn3)C2)C)=O)CC2CCC1C2 25599,CS(=O)c1ccccc1C(=O)NC1C=CC(CNC(=O)Cc2ccns2)C1 25600,C(CC(CC)(CC)NC(=O)C(C)NC=O)NC(c1cn(CCC)nn1)=O 25601,c1(NC(=O)NCCC2(C#N)CC2)ccc(C(F)(F)F)cc1Cl 25602,C=CC1(C(N2CCC(OC(C)C)CC2)=O)CCN(C(=O)C(CC)N(C)C)C1 25603,Cc1cc(C(N2CCCC2CNC(C2(C3CCC3)CCC2)=O)=O)nc(C)n1 25604,c1(C(N2CCN(C(CCSCc3ccc(C)cc3)=O)CC2)=O)cnc(F)cc1C 25605,c1(CNCC(CC)(C)C(N)=O)ccc(Cl)c(Cl)c1.C12(C)CC3CC1CC3O2 25606,c1(NC(N2C(CC(=O)NC3CCC(CO)CC3)COCC2)=O)cnnc(Cl)c1Cl 25607,C1(NC(CC2CC(C)N(C(=O)CC3CCSCC3)C2)=O)CCCC(O)CC1 25608,CCC(C)C(C(=O)N1CCCC1(C)C(=O)NCCSC(F)F)N(C)C 25609,c1(-c2c(COC)noc2)nc(Cn2nccn2)nn1Cc1cccnc1 25610,c1(CC(N2CC(CC(C)NC(c3c(CCC)n[nH]c3)=O)C2)=O)cnccc1OC 25611,c1(OC)cc(C(=O)NCCCCNC(=O)C(F)Cc2ccccc2)c(O)c(Cl)c1 25612,c1(OCC)c(OC)cc(C(=O)NC2CCN(C(=O)C(F)F)CC2F)cc1Cl 25613,C1(NC(C2CCN(C(CC)=O)CC2)=O)CN(C(=O)Cn2cc(Cl)cn2)C(C)(C)C1 25614,N1(C(c2c(C)scn2)=O)CC(C)CN(C(c2ncncc2Cl)=O)C(C)C1 25615,N#Cc1cc(C(N2CC(NC(C3CC(F)(CO)C3)=O)C(C3CC3)C2)=O)ccc1F 25616,N1(C(CC(=O)NC)=O)CCC(NC(=O)CSCCc2ccccc2)C1C 25617,c1(C(=O)Nc2ccc(CC)cc2O)cccc2occc12.c12nc(sc1C)C2 25618,Cc1cc(C(=O)NC(C2CCCN(c3nnc(CO)s3)C2)C)nn1C(C)C 25619,C1(N(C(CC(C)C2CCCO2)=O)C)CCC(CNC(=O)CCc2cccs2)CC1 25620,N1(C(C(CCC=C)(F)F)=O)CCC2(CC1)COC(CNC(=O)CN(C)C(C)C)C2 25621,c1(C(=O)NC(C2CC2NCc2cccc(C(F)(F)F)n2)=O)cc2ncccc2o1 25622,C1(CNC(C2(C)CC3CC3C2)=O)CCCCN(C(=O)COCC2CC2)C1 25623,CCS(=O)c1ccccc1C(N1CCCN(CCNC(C2CC2C)=O)CC1)=O 25624,N1(C(c2n(C)ncc2)=O)CCC2(CC1)CC(NC(=O)C(C)(CO)CO)CO2 25625,C1(NC(c2cc(C)sc2)=O)CCCN(C(=O)CN2CCC(=O)NC2=O)CC1F 25626,Cc1nc(N)c(CC(=O)NCC(C)(O)CNC(=O)CC(C)N(C)C)c(O)n1 25627,Cc1nc2cc(C(=O)NCC(CNC(c3cn(C)cn3)=O)CO)cnc2[nH]1 25628,c1(C(=O)NC2C=CC(CC(=O)N(C(C)C)CCN(C)C)C2)cccc(C#N)c1F 25629,C(C)(CNC(C1(C2(C)OCCO2)CC1)=O)(CC)NC(C1C(=C)CC1)=O 25630,N1(CC)CCCN(C(c2ccccc2C(F)(F)F)C(=O)NC2CCOC2)CC1 25631,Cc1cc(F)cc2[nH]c(C(=O)NCCCCC(C)NC(=O)C(N)=O)cc12 25632,c1(OCC(=O)NC(C2CN(C(CNC(C)=O)=O)C2)C)cccc2ccccc12 25633,n1(CC)cnc2c(N(CC(C)(C)C)C)[nH]c(=NC3CCOC(C)(C)C3)nc12 25634,Cc1ccn2c(C(=O)NCCCNC(c3cccc(O)c3Cl)=O)cnc2c1C 25635,N1(C(C(C)N(C(CC(C)OCC)=O)C)=O)CCN(C(=O)CO)CC1 25636,C1(NC(C2C(C3C(C)C3)C2)=O)CCN(C(=O)Cc2ccccc2Br)C1(C)C 25637,n1(CC(=O)NCC2(NC(C=CC)=O)CC3CCC2C3)cc([N+](=O)[O-])ccc1=O 25638,Cc1ccccc1OCC(=O)NC1CN(C(=O)CCC2NC(=O)NC2=O)CC1O 25639,c1(CC(=O)N(C2CC(NC(C3CC34CCCC4)=O)C2)C)c[nH]c2ccc(Cl)cc12 25640,c1(C(=O)NCCC(C)NC(C2COC(=O)N2C)=O)ccc(SC(F)(F)F)cc1 25641,C1(C(=O)NCCCN(C(C(C)SC)=O)C(C)C)CC(=O)N(c2ccccc2)C1 25642,N1(C(C)=O)CC2CC1CN2C(C1CC(N(C)C(C2C3CCC(=O)C23)=O)C1)=O 25643,C(=O)(CC(C)C(=O)OC(c1cc(Cl)no1)C)OC 25644,C(=O)(C1=C(Cl)CCC1)N(CCC)CCNC(=O)CNC(c1cnccn1)=O 25645,N1(C(C=C2CCC(C)C2)=O)CCC(C2(NC(c3cc(F)c(F)c(F)c3)=O)CC2)C1 25646,c1(CC(=O)NC)ccccc1NC(=O)NCC1CC(C)OC1C 25647,N1(Cc2cn(CCCCCN)nn2)CCOc2ncccc21 25648,C1(CNC(COCCC#C)=O)CC(C)N(C(=O)CCc2cncc(F)c2)C1 25649,CC(CC(=O)N1CCN(CC(N2CC(F)(F)CCC2C)=O)CC1)C(C)(C)C 25650,c1(C(=O)OC)cc(C)cnc1N(CC(O)CNC(=O)C(=Cc1cccnc1)F)C 25651,c1(C(N(C)CC2CCC2(F)F)=O)cnc(N(C)C)nc1 25652,C(CN=C(NCc1c(Br)nnn1C)NC1CCN(C2CCCC2)C1)OCC 25653,C1(CNC(C2(CCCC)CC2)=O)CCCCCN1C(c1ccccc1OC)=O 25654,CN1CC(C)(C)CC1C(N1CC(C2CCN(C(=O)CSCC(F)(F)F)CC2)C1)=O 25655,Cc1cc(O)c(C(=O)NCCCN(C(=O)COCCCF)C)cc1Br 25656,C(CC(F)F)(C(=O)N(CC)CC1CCOC1)NC(C=CCC)=O 25657,C=CCN=C(NCc1ccc(F)cc1)NC1CCCN(CC(F)F)C1 25658,N1(C(C2C(C(C)C)C2)=O)CC2CN(C(=O)C3=CCCC(C)(C)C3)CC2C(F)(F)C1 25659,N1(C(=O)CCc2ccoc2)CC2CN(C(c3ncc(Cl)s3)=O)CC2C1 25660,Cc1ncnc(C(N2CCC(CN(C)C(c3n[nH]cc3C(F)(F)F)=O)C2)=O)c1C 25661,N1(C(=O)CSCC(F)(F)F)CCC(C(=O)NCC2(O)CCSC2)C12CCC2 25662,N1(C(C(C)NC(C)=O)=O)CCC(C2OCCC2NC(c2ccns2)=O)CC1 25663,C(C(F)(F)F)(C1CCCCC1)NC(=O)NC(c1cscn1)C 25664,N1(C(C(C)(C)C2CCOC2)=O)CC2C(CNC(=O)C(N)=O)C2C1 25665,Cc1ccc(C=CC(=O)NCC(O)CN(C(=O)CN2CCCCC2)C)c(C)c1 25666,c1(C(=O)NCCN(C(C=C(CCN(C)C)Cl)=O)C2CC2)cnc(CC2CC2)nc1 25667,C1(F)(CNC(=O)CC2(O)CCCCC2)CCN(C(=O)CCNc2ccccc2)C1 25668,C(=O)(C(C)C1=CCCC1)NCC1CN(C(COCCCC)=O)CC12CC2 25669,CC(C)CC(CCO)NC(=O)CC1CN(C(C2(O)CCCCCC2)=O)CC1C 25670,C1(O)(C(C)CNC(=O)CSC(F)(F)F)CCN(C(c2scnc2C2CC2)=O)C1 25671,CC1CN(C(=O)C(C2(O)CCC2)NC(c2cncc(CO)c2)=O)CCS1=O 25672,C(CNC(c1ccc(N2CCC(C)(C)C2)cc1)=O)(CCS(C)(=O)=O)OC 25673,C1(C(N2CC3C(CNC(CNC(C(C)(C)C)=O)=O)C3C2)=O)CC2(CCOCC2)C1 25674,C1(C(N2CC(NC(=O)COc3cn[nH]c3)C2)=O)(CSC)CCC1 25675,C(=O)(C1=NOC(CC(=O)C=O)C1)Nc1ccccc1.C1(N)CCC(OC(F)F)C1 25676,C(=O)(CCCC(=O)NCCN(C(=O)CCS(=O)(=O)N(C)C)CC)NCCC 25677,C(C1CCCCC1)=CC(=O)NC1(C2N(C(C3CC(N(C)CC)C3)=O)CCC2)CC1 25678,N1(Cc2ccc(C(=O)OC)[nH]2)CC2CCN(C(c3ccc(C#N)s3)=O)CC2C1 25679,c1(OC)ccccc1-n1nnnc1C(c1c(I)cnn1C)Nc1cnoc1 25680,c1(C(=O)NCC2N(C(CCC)=O)CCCC2C)cc2ccccn2c1 25681,Cc1cc(C(N2CC3CC2CC3NC(=O)C2=COCCC2)=O)c(S(N)(=O)=O)s1 25682,N1(C(c2cc(C)c(C(N)=O)cn2)=O)CC2CCC1C(CNC(C1(CO)CC1)=O)C2 25683,c1(C(C)C)cccc(CNC(c2cnccc2Cl)c2nnnn2CC2(C)CC2)c1 25684,N1(C(c2sc(C)c(O)n2)=O)CC2COCCC2(NC(C2OCC3CCCC23)=O)C1 25685,c1(C(C)C(=O)NC2CCC(NC(C3CC(Cl)(Cl)C3)=O)CC2)ccc(C#N)cc1 25686,Cc1ccc(F)c(C(=O)NCc2occc2C(=O)NC(C)C(F)(F)F)n1 25687,C1(N(C(=O)CN2CCS(=O)CC2)C)CN(C(C2CCCCCC2)=O)CC12CC2 25688,C=CCC(C(=O)NC(C)CC(C)(C)OC)NC(C1(CO)CCCCC1)=O 25689,c1(C(=O)NCCC(CCNC(C(CCSC)O)=O)C)ccc(=O)n(CC(C)O)c1 25690,S(=O)(=O)(c1cccc(=NCC2CCC3CC23)[nH]1)NCCC(CC)(C)C 25691,c1(C(N2C(CNC(c3c(C)cco3)=O)CN(C)CC2)=O)ccc2nccn2n1 25692,C1(C(=O)NC(CCOC)CNC(=O)CC2(OC)CCC2)Cc2nccn2C1 25693,Cc1nn(C)c(C)c1C(=O)C(=O)NC(CNC(c1cc[nH]c(=N)c1)=O)C(C)(C)C 25694,Cc1oc(S(N)(=O)=O)cc1C(N1CCC(NC(C2CC2C(N)=O)=O)CC1)=O 25695,CC(CCCO)N=c1[nH]c2c(c(=NCC3OCCC3C)[nH]1)COC2 25696,Cc1cc(C(=O)NC2CC3(C2)CC3NC(c2cscc2Cl)=O)cc(C)c1Cl 25697,c1(CC(=O)N(C)CC2CCN(C(c3c(CC)ncs3)=O)C2)cccc(F)c1O 25698,C1(CC(=O)N(CC(C)(C)NC(c2c(C)con2)=O)C)CCOC(C(C)C)C1 25699,C1(OC(=O)CC2SC3=NCCN3C2=O)C=C(c2ccc(Cl)cc2)CCC1 25700,CCCC(CCCNC(C1CCCCC1O)=O)NC(c1cc(C(C)C)no1)=O 25701,C1(NC(c2n(CC)ccc2)=O)(CF)CCN(C(=O)C=C(C)C(C)C)C1 25702,N1(CC)CC(NC(C2(CNC(C3CCC=CCC3)=O)CCC2)=O)C(C)C1 25703,c1(C(=O)NCCNC(CCc2c(C)nn(C)c2C)=O)nc(=N)[nH]c2ccccc12 25704,C(C(=O)Nn1cnnc1C)C1CN(C(Cc2c(C)con2)=O)C(C)(C)C1 25705,C(C(CC(C)C)C(=O)N(C1CCCC1O)C)NC(c1cc(C)oc1)=O 25706,C1(OCCNC(C2C(C)CCS2)=O)CCN(C(=O)CCOCCCN(C)C)CC1 25707,C1(CNC(=O)C=Cc2cccs2)CCN(C(c2cn(C(F)F)cn2)=O)CC1 25708,c1(CCC(=O)NC2(C)CC(NC(COCC)=O)C2)ccc(C#N)cc1 25709,C(=O)(CCC(C)(C)N(C)C)N1C(CNC(c2ncc(OC)cn2)=O)CC1 25710,N1(C(CNC(=N)N)=O)CC2(CCCC2NC(=O)Cc2c(Cl)cccc2Cl)C1 25711,C1(CNC(c2c(C)nn[nH]2)=O)CC(O)CN1C(=O)CCCCN(C)C 25712,c1(OC)ccc(Cc2csnc2CNC(=O)NCC2CCC2C2CCCN2)cc1 25713,C1(CNC(CC(C)SC)=O)CN(C(C2CC=CCO2)=O)CCC1C 25714,CCCCC(CC(=O)NC1CC2(C1)CC2(F)F)NC(c1cccc(O)c1F)=O 25715,CC1CCN(C(=O)C=CCO)C(C)C1NC(c1cc(C(F)F)[nH]n1)=O 25716,C(c1cc2ccccc2o1)=CC(N1CCC(CN(C(CN(CCC)C)=O)C)C1)=O 25717,c1(C(=O)NCC(CC=C)NC(C2CC(O)CN2C)=O)c(F)ccc(C)c1Cl 25718,N1(C(C(C2CCOCC2)OC)=O)CCC(CCCCNC(=O)CSC)CC1 25719,c1(OC)cnc(C(F)(F)F)cc1C(=O)NC1(C)CN(C(=O)C(O)Cn2cncn2)C1 25720,N1(CC(=O)NC2CCC(C(=O)NC(COC)COC)C2)C(=O)CCC1=O 25721,C=C(C(=O)NC1CC1C(=O)Nc1cc(F)ccn1)C(F)(F)F 25722,c1(C(=O)NCCN(CC(C)O)C(=O)C=Cc2cnccn2)cc(O)cc(C#N)c1 25723,Cc1ccc(C)c(C(N2CC3C(CN(C)C(C4(c5cccs5)CC4)=O)C3C2)=O)n1 25724,C1(C(=O)NCc2ccc(CC(=O)O)cc2)CN(C(C2(F)CCC2)=O)CC1(F)F 25725,CC1CN(C(=O)C(N2C(C)CCC2C)C)CCN1C(=O)CCCC(C)O 25726,CCCC(CCC)=Cc1nc(C2(C(=O)N(C)C)CC2)no1 25727,N1(C(COC)=O)CCC12CN(C(=O)C(CC(C)C)NC(=O)CNC(=O)C(=O)O)C2 25728,CN1C(=O)OC2CN(C(C3(F)CN(C(c4ccncc4Cl)=O)C3)=O)CC12 25729,N1(C(CCC#C)=O)CC(N(C(=O)C(C)N(C)C)C)C2(CC2)C1 25730,N1(C(CSCC#C)=O)CC(C(N2CCc3nc[nH]c3C2)=O)CC(C)(C)C1 25731,C1(C(N(CCN(C(CCOCCCOC)=O)C(C)C)C)=O)CCC(N=[N+]=[N-])CC1 25732,N1(C(C2CCC(=C)CC2)=O)CCC2(CC(NC(=O)CCOCC(C)C)C2)C1 25733,C=CC1COCC1NC(=O)C(O)CCNC(=O)CCOCC(F)F 25734,CC(C)CC(C(=O)NCC1C2CCOCC12)N(S(C)(=O)=O)C1CC1 25735,c1(NCC2(CCC)CC2)nc2ccccc2nc1NCc1cc(Br)ccc1N 25736,C12(c3onc(C)n3)COC(CN1CC(=O)N(CCn1ccnc1)Cc1ccccc1)C2 25737,c1(C(C)=O)ccc(C(=O)NCC=CCC(=O)NCCCCCC)[nH]1 25738,C(CC(N)=O)(C(=O)N1CCCC1CC(N)=O)NC(C(C)n1ccnn1)=O 25739,C1(NC(c2occ(C)c2)=O)CCCCCCC1NC(c1cnn(C2CC2)c1)=O 25740,c1(C(C)O)ncc(C(N2CCC2CNC(=O)C(C)OC2CCCCC2)=O)s1 25741,O(NC(=O)C(CNC(=O)Cn1ccnn1)N(C)C)C(CC)C 25742,C(C(CC)(CC)C(=O)NC1CCN(C(C)=O)CC1C)NC(Cc1cn(CC)nn1)=O 25743,C1(C(=O)Nc2cncc3nc(C)[nH]c32)CC(N=c2nc(C#N)[nH]cc2Cl)C1 25744,N1(C(C=NOC)=O)CC2CCC1C1CN(C(=O)CCn3cc[nH]c(=O)c3=O)CC21 25745,CN1C(=O)NCC1C(=O)NC(C1CCCC1)CNC(=O)C=CC1CCOC1 25746,C#CCCC(O)C(=O)N(C1CN(C(=O)C2=CSCCO2)C1)C 25747,O(P(=O)(OCC)C1(NC(C2(F)CCOCC2)=O)CNC1)CC 25748,Nc1nccnc1C(=O)NCC(c1ccccc1)CNC(C1COCC1CF)=O 25749,CC1C(NC(C2CN(C)C(=O)N2)=O)CC2CCC1N2C(c1ccsc1C(F)F)=O 25750,c1(CC(=O)N(C(C)CN(C)C(C2CC(O)C2)=O)C)ccc(F)nc1 25751,c1(C(N2CCCC(NC(C3(C)CCN(C(C)=O)C3)=O)C2)=O)ccn2ncccc12 25752,C1(OC)CC2CCC1(N)C2.C1(F)(F)C(=O)C12CC2.c1(Cc2cnoc2)cn(C)nn1 25753,N1(CCNC(C2(NC(CCO)C3CCCC3)CCCO2)=O)CCCCC1 25754,C(COC)(C(=O)N(c1ccccn1)C)NC(COC)=O 25755,N1(C(CN(C(C(C)OCC2CC2)=O)C2CCC2)=O)CCC(O)C(C)(C)C1 25756,c1(C(N2CCCC(F)(CNC(c3ccncc3F)=O)C2)=O)cccc2nn[nH]c12 25757,Cc1nc(C(=O)NCC(c2ccccc2F)NC(=O)C=CC2CCCC2)c(C)s1 25758,N1(C(C=C(C)C2CC2)=O)CCOC(C)(CNC(c2ccc(Cl)s2)=O)C1 25759,N1(C(c2cccc(I)c2)C(=O)NCCOC)CCCC(O)(c2ccccc2)CC1 25760,n1(CC)ncc2cc(C(=O)NC(CNC(c3nocc3Cl)=O)CC(C)C)cnc12 25761,c1(-c2nc(C(CC)CC)nn2Cc2cccs2)cnc2n1CCCCC2 25762,C(CCC(=O)N1CCC(C(C)NC(C2(CC)CC2)=O)C1)NC(=O)OCC 25763,C#CCCCCC(=O)N1CCC(C(F)(F)F)C(NC(c2cccnc2C)=O)C1 25764,C1(NC(c2ccccc2Br)C(=O)O)CCN(CC(F)(F)F)C2(CC2)C1 25765,CCCC(C(=O)NCc1cc(C)ns1)NC(=O)CC1CCOC1(C)C 25766,C1(CNC(C(C=C)C)=O)CC(C(=O)N(CC(C)O)C(C)C)=NO1 25767,CCCC(CCC)CC(=O)NC(C(=O)NCC(F)Br)C1(O)CCC1 25768,c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)C2)nc2ccccc2[nH]1 25769,c1(C(=O)Nc2cc(C(=O)OC)c(C)nc2)cc2c(=O)n(C)c(=O)n(C)c2s1 25770,N1(C(C(CCO)N(C)C)=O)CC(NC(c2ccc(O)nn2)=O)C(C2CC2)C1 25771,c1(C(=O)NCC2C(C)(C)C(NC(=O)Cc3cc(Cl)cs3)C2)ccc2c(c1)CC2 25772,C1(C(=O)NC2C(NC(c3c(C)c(N)ccc3)=O)COCC2)CC2(C1)CC1(CC1)C2 25773,N1(C(CCC2C(C)(C)C2)=O)CCC(OCCNC(c2sccc2F)=O)C1 25774,C1(NC(C2CC(C)CC(C)C2)=O)CCOC12CCN(C(=O)OC(C)(C)C)CC2 25775,C1(C(=O)O)CN(C(=O)NCCc2cnco2)C2(CCC2)C1 25776,c1(C(=O)NCCC2(CNC(C3C(C)(C)CC3)=O)CC2)cccc(OC(F)F)n1 25777,C(CCN=c1[nH]c(=NCC2COC(C)(C)CO2)[nH]c2c1CSC2)NC(C)=O 25778,c1(C(N(CC)CC2CCCN2C(c2occc2F)=O)=O)[nH]c(O)nc1C 25779,c1(N2CC=CCC2)nc(=NCC2CN(S(C)(=O)=O)C2)[nH]c2c1CSC2 25780,c1(C(N(CC(CC)NC(=O)CSC(F)F)C)=O)ccc(-c2ccncc2)s1 25781,c1(C(N2CCN(C(c3c(OC)csc3)=O)C(CO)C2)=O)cn2ncccc2n1 25782,C(=O)(C(C)(C)Nc1ccccn1)NCCCN(C(=O)CN1CC(C)(C)C1)C 25783,N1(CCNC(C(C)(C2(C)CC2)OC)=O)CCC(NC(C2CN(C(N)=O)C2)=O)CC1 25784,Cc1nc2c(C(=O)NCC3CCCN3C(=O)C=Cc3sccc3C)cccc2o1 25785,c1(OC)ncc(Br)cc1CN1CCC(CC(=O)NCCCC(F)(F)F)CC1 25786,c1(CC2N(CCC(=O)OC)CCC2C)ncc(C)cc1Cl 25787,Cc1cccc(C(C(C)C)NC(c2cccc(C(=O)O)c2)=O)c1 25788,C1(CNC(=O)CO)CN(C(=O)COc2ccccn2)CC1(F)F.CC1C(=O)O1 25789,N1(C(C2CCCC(=O)C2)=O)CC=C(C(=O)NCC(c2cccnc2)O)CC1 25790,CCCCC(C(=O)Nn1cnnc1C)NC(c1ccc(C#N)s1)=O 25791,CC1=C(C(=O)NC(CCN(C(=O)CC2CCCC23CC3)C)C(C)(C)C)CCO1 25792,CC1CCN(C(c2cc(Cl)nnc2O)=O)CCN1C(C1CC1C1CCCC1)=O 25793,N1(C(CC(C=C)C)=O)CCCC(O)(CNC(=O)COCc2nccs2)C1 25794,N1(C(C(=Cc2cccnc2)C)=O)CC(NC(=O)CCCNC(N)=O)CCC1C 25795,C(=O)(C(O)CC(C)(C)C)N1CC(CNC(C(C(=O)OC(C)(C)C)OC)=O)(OC)C1 25796,Cn1cc2c(C(=O)NC3CCCN(C(=O)CCc4nc(=N)[nH][nH]4)C3)cccc2n1 25797,CC1CC(CCNC(c2cccs2)CO)C1 25798,C(N=c1[nH]c2c(c(=NC3CCC4CCC34)[nH]1)CCCC2)c1cc(COC)on1 25799,c12ccc(s1)C=CC(=O)NC1(CC1)CCN2.C(=O)(COC)NCC1CCC1.CC=C 25800,S(=O)(=O)(c1ccc(NC2CCN(c3cn(C)nc3Br)C2)nc1)N(CC=C)C 25801,n1(CC(=O)O)cc(CSCC(=O)NC2CCN(C(=O)CC3CCCO3)C2)nn1 25802,N1(CCNC(C2(CNC(C3CS(=O)C3)=O)CCC2)=O)C(=O)CNC1=O 25803,Cc1nc2ccsc2c(=NCC2CCCCN2C(C2CC3(C2)CC(F)(F)C3)=O)[nH]1 25804,C1(C(=O)NCC(O)CNC(C2CN(C(C)=O)CC2OC)=O)(COC)CCCCC1 25805,N1(Cc2cccc(C#N)n2)Cc2ccc(NC(C3CC(O)CN3)=O)cc2C1 25806,C1(N(C(C(C(=C)C)(C)C)=O)C)CC2CCC(C1)N2C(=O)C1=CC2CCCC12 25807,CCC(CC)CCC(=O)N1CCOC(C(C)NC(=O)C#CC2CCC2)C1 25808,N1(C(C(N2CCC(c3nc(=N)[nH][nH]3)C2)=O)=O)CCC2(CC1)CC2C(=O)O 25809,N1(C(C(CCOCC)NC(c2ccns2)=O)=O)CC2C3CCC(O3)C2C1 25810,C1(NC(C23OCC(CC)(C2)C3)=O)CCN(C(c2cc(Cl)c(Cl)s2)=O)CC1F 25811,C1(C2CCC2)(NC(C2CCCC(C(=O)O)C2)C)CC1 25812,C1(C(=O)NCCCC(C)NC(=O)Cc2cccc(F)c2)COCC2(CCC2)O1 25813,N1(C(c2c(C)sc(Cl)n2)=O)CCN(C(c2ncc[nH]2)=O)CC(O)C1 25814,N1(C(=O)CCC=Cc2ccccc2)CCN(C(=O)Cn2cc(Cl)cn2)CC(O)C1 25815,c1(C(=O)Nc2cc(F)ccc2F)n[nH]c2c1CN(C(C1(F)CC1)=O)CC2 25816,C1(C(=O)NCc2cc(=N)[nH]cn2)(COC)Cc2ccccc2C1 25817,CCCCCC(=O)NCCC1CC(NC(c2cc(-c3cccc(O)c3)on2)=O)C1 25818,c1(C(=O)NC2CCCN(C(C=Cc3ccc(C)s3)=O)C2)ccc(F)c2occc12 25819,c1(C(C)=O)cc(C(N2CCC(F)(CNC(c3cnnn3C)=O)C2)=O)oc1C 25820,c1(OC)cncnc1C(N1CC2C(CNC(=O)CCC3CCCCO3)C2C1)=O 25821,N1(C(c2c(C)cc(CC)o2)=O)CC(C)CCC1C(=O)NCc1nncn1C(C)C 25822,N1(C(c2n(C)nnc2)=O)CCCC1C1CCCCN1C(=O)CCn1ccnc1 25823,CCS(=O)CC(=O)NCCCC(C)(C)NC(=O)C(C)NC(c1ccoc1)=O 25824,CC1CN(C(=O)CCc2ncc[nH]2)CCCN1C(c1cncc(CO)c1)=O 25825,CN1CCN(C(c2c(C3CCC3)cnn2C)=O)CC1CNC(=O)C1=CCOC1 25826,c1(C(N2CC(C(C)NC(c3c(C)ccnc3O)=O)C2)=O)cccc2[nH]ccc12 25827,C(C)(c1ccc(OC)cc1)=CC(=O)N(C1CCCN(C(CC(CCC)O)=O)C1)C 25828,C1(CNC(C(=O)NCC(F)F)=O)CCN(C(C23CC(CO)(C2)C3)=O)C12CCC2 25829,Cc1cc(C2CCCO2)cc(C(=O)NC(CNC2(C3(C)CC3)CC2)CC(C)C)n1 25830,c1(CC)cc(C(=O)NC2CC(NC(c3nn(C)cc3N)=O)CC2O)n(C)n1 25831,c1(C(=O)NC(CC)CN(C)C(C2(c3ccc(F)cc3)CCC2)=O)[nH]ncc1C#N 25832,N1(C(C2CC(=O)N(Cc3ccc(Cl)cc3)C2)=O)C2CCC1CC1(C2)CC1(F)F 25833,c1(CC(=O)NC2C(NC(Cc3nnc(C)o3)=O)CCCC2)cccc(O)c1F 25834,CCCS(=O)(=O)CC(=O)N(CC)CC1CCN(C(C2(F)CC2C)=O)CC1 25835,CC(CS(C)=O)C(=O)NCCOCCNC(c1cc(N)cc(O)c1)=O 25836,c1(C(=O)NC23C(CN(C(CSC)=O)C2)C3)c(Cl)oc2ccccc12 25837,C(=O)(CCCCCC#N)NC(C)CC(C)NC(c1cccc(OC(F)F)c1)=O 25838,C(=O)(C1=C(Cl)CCOC1)N1CCC(C(=O)NCC(CC)C(C)(F)F)C1 25839,C(=O)(CC(C)(C)O)NCC(C)NC(C1(n2cncn2)CC1)=O 25840,CC1(C)CC(NC(=O)CCC2CCOCC2)CN1C(=O)CN1CCCCCC1 25841,N1(C(c2nc(C)oc2)=O)CCN(Cc2cc(Br)ccc2I)C(C)C1 25842,C1(C(C(C)C)NC(=O)C(Cl)=CCl)CN(C(=O)C=Cc2cn(C)cn2)CCO1 25843,n1(CCC(=O)NC(CNC(=O)C(C2CCCCC2)F)C2CC2)cnc([N+](=O)[O-])c1 25844,C1(C(C)NC(C(C)(C)OC)=O)CCCN(C(=O)CC(C)(F)F)C1 25845,C=CCCC(C(=O)NC(C(N)=O)C1CCCC1)NC(c1cc(Cl)n[nH]1)=O 25846,Cc1cc(C(=O)NCCC(C)NC(C2CNC(=O)C2)=O)c(Cl)cc1F 25847,c1(C(N2CC(CCNC(C(CCCC)C)=O)C(C)C2)=O)nccn2cc(C)nc12 25848,N1(C(c2cc(OC)cc(CC)c2)C(=O)OCC2CC2)CC2C3C=CC(O3)C2C1 25849,C1(c2nnc(C)o2)CN(C(CC2CCC3CC23)C(=O)NC2COC2)CCO1 25850,N1(C(CCCC#C)=O)CC2(C1)CN(C(c1cccc(C(F)(F)F)c1Br)=O)C2 25851,C1(C)(NC(C(C2CN(C(c3cccc(CC)n3)=O)C2)OC)=O)CCCCC1C 25852,C1(NC(C(=Cc2ccncc2)C)=O)CS(=O)(=O)CC1NC(c1cnc[nH]1)=O 25853,Nc1cc(F)ccc1C(=O)NC1CCCN(C(=O)C(O)CN2CCOCC2)CC1 25854,C1(NC(c2c(CC)nc(C)nc2)=O)C(C)CCN(C(=O)Cc2cn(C)nn2)C1C 25855,CS(=O)(=O)CC(=O)NC1CCOC(C(=O)NOCC(=O)OC(C)(C)C)C1 25856,N1(C(CC(CC)(F)F)=O)Cc2nccn2CC(NC(=O)C(F)C(C)C)C1 25857,c1(C(=O)NC2CCCCCN(C(CC=C)=O)C2)n[nH]c2cc(Br)ccc12 25858,Cn1cnc(I)c1C(N1CCC(c2ccncc2)CC1)C(=O)NC1CCOC1 25859,Cc1cncc(C=CC(=O)N(C)CCC2CCN(C(=O)CCS(C)(=O)=O)CC2)c1 25860,Cc1[nH]nc(C(=O)N(C)CC2CN(C(c3ocnc3C(F)(F)F)=O)CCO2)c1F 25861,C(=O)(CCCC(C)O)NCC(C)(C)Nc1nccc(CC(=O)OC)n1 25862,N1(C(c2cc(COC)no2)=O)CC2CN(C(=O)C(C)CS(C)(=O)=O)CC2C1 25863,c1(C(=O)NCC2CC(C)(C)CN2C(=O)Cn2cnc(=N)[nH]2)cc2c[nH]cnc-2n1 25864,Cc1c(C(N2CCC2CNC(=O)C(F)CC(C)C)=O)sc2[nH]cnc(=S)c12 25865,c1(C(=O)NC(CN(C(c2c[nH]cc(Cl)c2=O)=O)CC)C)n[nH]c2cc(Cl)ccc12 25866,N1(C(CCOC)=O)CCC(NC(c2cc(C(C)C)n(C)n2)=O)C1c1ccccc1 25867,N1(C(COCC(=O)OC)=O)CC2CC1C2NC(=O)C(C)(C)n1ccc(C2CC2)n1 25868,CC1CCn2cc(C(=O)NCC(CO)NC(c3c[nH]c(Br)c3)=O)nc2C1 25869,N1(C(c2ccc(CO)nc2)=O)CC=CC(C(N2C(CO)CCC2CO)=O)C1 25870,CCCCS(=O)(=O)CC(=O)NCCCN1CCN(C(=O)C2=CS(=O)CCC2)CC1 25871,C#Cc1ccc(C(=O)NC2CCN(C(c3c(C)ncn3C)=O)CC2O)c(OC)c1 25872,C1(CNC(C2CN(C(N)=O)C2)=O)CN(C(c2cc(F)ccc2Cl)=O)CC12CC2 25873,C1(C(=O)NCC(C)(C)N)C2CC2CN1C(=O)C(C)OC.C(C(C)C)O 25874,Cc1ncsc1C(=O)NCCOCCC(=O)N(C)CCc1cnc[nH]1 25875,N(C1COc2ccccc21)CCOC(C)C(=O)NC(CCSC)C(=O)NCC.CO 25876,c1(C(C)(C)C)cccc(C(c2nnnn2C2CCCC2)NCCc2cccs2)c1 25877,N1(C(C)C(=O)NC(=O)NC(C)(C)C)CCCC(C(=O)Nc2cc(O)n(C)n2)C1 25878,N12CCCC(C1)C2=O.Cc1ncsc1CCNC(=O)NC(C)C 25879,C(C)(C)(C#CCCC)NC(CCN(CC#C)C(C1CCCC(O)C1)=O)=O 25880,C(C)(CCCCNC(C12CC(C)(C1)C2)=O)NC(c1c(C)ocn1)=O 25881,C1(C(N(C)CCNC(c2sncc2Br)=O)=O)CN2CCC1CC2 25882,c1(NC(C2C(NC(c3ccc(C)s3)=O)CC2)=O)cc(F)c(O)cc1C 25883,Cc1cccc(NC(=O)NCC(=O)NCCNC(=O)CC2CCC2(C)C)c1 25884,C12CCOC(C1)C(=O)N2.C1(CCCC)(NC(=O)NCCC(=O)OC)CCCC1 25885,N1(C(CCCS(C)(=O)=O)=O)CCC2(CC1)CCN(c1ncnc(=N)[nH]1)C2 25886,c1(C(=O)NC(C2CN(C(=O)CCCCC(N)=O)CCO2)C)cc(Cl)c(F)cc1F 25887,c1(NC(C(C)(C)CCl)=O)ccn2c(C(F)(F)F)nnc2c1 25888,c1(C(=O)NC2CCCCN(C(CC(=C=C)C)=O)C2)c(F)cc(O)cc1F 25889,c1(C(N2CCC(N(C(=O)C3=CC(C)(C)C3)CC)C2)=O)ccc2c(c1)C(=O)NC2=O 25890,c1(OCCC(=O)NC2(CC=C)CCN(C(=O)CSC)C2)cc(Cl)ccc1Cl 25891,N1(C(CNN2C3CC(N)C2CC3)=O)CC(=O)Nc2ccccc21 25892,c1(CC)nn(C)cc1C(=O)NCC=C1CCN(C(C2(OC)CCCC2)=O)CC1 25893,c1(OC)ccc(F)c(C(=O)NC2CC3CCC2(NC(c2nccc(C)n2)=O)C3)c1 25894,C1(NC(CCc2c(C)noc2)=O)CC(C)N(c2nc(-c3ccccc3)ns2)C1 25895,N1(C(C2C(NC(=O)Cc3ccccn3)C=CCC2)=O)CC(O)C(O)C1CO 25896,S(=O)(=O)(c1ccccc1)NCC(=O)N(CC(CC)NC(=O)C(C)N(C)C)CC 25897,c1(C(=O)NC(CNC(C(C)C2CC2)=O)(C)C2CCC2)cc(-c2cnn(C)c2)on1 25898,c1(OCC(=O)NCC2CC(NC(c3cc(C)oc3)=O)C2)ccc(S(N)(=O)=O)cc1 25899,C12CN(CC1(C)C)C2=O.c1(C(N(C(CC)C)C)=O)ccc(O)nc1Cl 25900,C1(NC(CCC2CCC(C(=O)OC)CC2)=O)CCN(C(C2(F)CC2)=O)CC1CO 25901,C(C(C)(C)CO)N(C(=O)C(CC1CCC1)NC(=O)C(C1CCCCC1)F)C 25902,N1(C(c2nnn(C)c2C(F)F)=O)C2CCC1CC(NC(=O)CCC1CC1)C2 25903,C(=O)(C1CCc2nccn21)NCCCCCCC(=O)N1CC(C)(C(=O)OC)C1 25904,C12(CNC(c3cc4ccncc4[nH]3)=O)CCC(CN(C(c3ccns3)=O)C1)C2 25905,C1(C(=O)NC2CCCN(C(CC)=O)C2)CC(C)CN(C(=O)CSCCC#N)C1 25906,c1(CO)c(O)ccnc1Sc1ccccc1-c1co[nH]c1=N 25907,c1(C(=O)NC(C)C(C)NC(=O)C(C)n2cccn2)cc2occc2s1 25908,C(=O)(C(CO)C(C)(C)C)N(C(CNC(CCCC=C)=O)C1CC1)C 25909,c1(OC)ccc(C(N2CC(F)CC2C(=O)Nc2ccnc(O)c2)=O)c(Br)n1 25910,C=CC(CCC)CC(=O)NC1C2CCN(C(=O)Cn3cnc(Br)c3)C12 25911,C(C(O)CC(=O)N(C)CC1(O)CCC1)NC(CNC(CC(C)C)=O)=O 25912,N#Cc1cnccc1N1CCCC1CNC(C1(CN2CCCC2)CC1)=O 25913,c1(C(N2CC(C)C2C(=O)N(C)CC2OCCC2(C)C)=O)cc2ccccn2c1 25914,c1(C(N(C)CCNC(C2(C)CCCC2O)=O)=O)c[nH]c(=NCC(F)(F)F)cn1 25915,Cc1oc(S(C)(=O)=O)cc1C(=O)NC(CO)C(C)NC(c1cnnn1C(C)C)=O 25916,N1(C(=O)CCc2cc(F)ccn2)CCC2C1CCN2C(=O)CCC12CC(F)(C1)C2 25917,c1(NC(c2c(CC)cc(Br)cc2)=O)ccc(S(=O)(=O)N2CCOCC2)cc1 25918,CC(C)CC(CNC(=O)C1=C(Cl)CCC1)C(=O)NC1CCCC(O)C1 25919,Cc1ccc2[nH]c(=NC(C)C3CCN(C(C4CCC=CCCC4)=O)CC3)sc2n1 25920,c1(CNC(CC(CC)C2CCC2)=O)cccc2c1CN(C(C1(CC)CC1)=O)C2 25921,N1(C(Cc2cc(C)cc(Cl)c2)=O)CCCc2c(O)cccc21 25922,C(=O)(CS(=O)(=O)C(C)(C)C)N1CCCC(C)(CNC(=O)CC(C)(O)C2CC2)C1 25923,c1(SC)ccc(C)c(C(N2CCCCC2CCN(C)C(c2nnc(C)s2)=O)=O)c1 25924,N1(C(C(C)OCC)=O)CCN(C2CCN(C(=O)C(O)COC)CC2)C(=O)C1 25925,Cc1ncc(CC(=O)NCC(C(C)C)NC(=O)C(C)CSC(F)(F)F)[nH]1 25926,c1(C(=O)Nc2cc(-n3cc(CC(O)CO)nn3)ccn2)c(F)cccc1Br 25927,N1(CCCCNC(c2ccc(C(C)C)c(F)c2F)=O)C(=O)c2ccccc2C1=O 25928,c1(NC(C2CCCC(NC(c3cccc(F)n3)=O)C2)=O)cc(Cl)ncc1[N+](=O)[O-] 25929,c1(C(N2CC(C)(C)C(CNC(c3nc(Cl)cs3)=O)C2)=O)ncnc2c1CCCC2 25930,CCCC(C)(C)CC(=O)NC(C1(O)CN(C(c2ccsc2SC)=O)C1)C 25931,Cc1ccc2cc(C(=O)NC3CCCN(C(c4ccn(C)c4)=O)C3)nn2c1 25932,C1(OC)CN(C(=O)CC2(O)CCOCC2)CC1NC(c1coc(C2CCC2)n1)=O 25933,c1(C(=O)NC2C(NC(CC(CC)C(C)C)=O)CCOC2)c[nH]c2cccc(Cl)c12 25934,CN1CC2C3CCC(C3)C2C(=O)N(c2cncc(C(F)F)c2)C1=O 25935,c1(CC(=O)NCC(CN(C(=O)COCC2CCCO2)C)O)sccc1Cl 25936,c1(C(N(CC(CN(C)C)O)C)=O)sccc1C1CC1.c12cnn(c1)CCNC2=O 25937,C1(NC(CN(C(=O)CC(C)n2cccc2)CCC)=O)CC12CCOCC2 25938,c1(NCC2CCC(=O)NC2)ccc(S(=O)(=O)NC(Cc2nccs2)CO)cn1 25939,c1(C(=O)NC(CCN(C(C(C)CC(N)=O)=O)C)C(C)(C)C)ccc2occc2c1 25940,CN1CC2CCC(OC(c3ccc(COc4ccccc4)cc3)=O)C2C1 25941,c1(C(C(=O)NCC(C)CNC(C2(F)CC2)=O)O)cnn(C)c1 25942,c1(C(=O)NC2CCCC(CNC(C(C)(F)F)=O)C2)ncc(C(N)=O)cc1Cl 25943,c1(SCC(=O)NCC(CCOC)NC(C2CCC(CO)CC2)=O)cccc(C)c1 25944,N12CC3CN(C3C1)C(=O)c1cnc(cn1)C2=O.c1(SC)cccc(N(C)C)c1 25945,c1(C(=O)NC2CC(C)SC2)c(CNC(c2cc(=N)[nH][nH]2)=O)cnn1C 25946,CCCC(C(=O)NC(C(=O)N1CCC(CC2CCC2)C1)C(C)OC)OCC 25947,C1(CN(C(C2(COC)CCOC2)=O)C)CCN(C(=O)CC(C)c2ccco2)CC1 25948,Brc1cc(I)c(CN2CCC(N3CCC3)CC2)s1 25949,n1(CC(N2C(CC(=O)NCc3ncc[nH]3)CC2)=O)ccc2ccccc12 25950,N1(C(c2cc(C)sc2C)=O)CC(N(C)C(c2cnc(N(C)C)s2)=O)C(C)(C)C1 25951,c1(CCCN2CC2)ccc(C(=O)O)cc1.C(CC(F)(F)Cl)SC 25952,Cc1nc(O)[nH]c1C(N1CC(C(N)=O)(CNC(=O)C(C)OC2CCCC2)C1)=O 25953,c1(OC)ccc(N2CCCCC2)cc1N1CCOC1=O.N12CCOC(C1)NC2=O 25954,Cc1nnc(CC(N2CC(NC(c3cnc(C)s3)=O)C2)=O)o1 25955,CC(CC1CCCO1)N=c1[nH]c(N(C)Cc2ccc(Br)s2)nc2ccsc12 25956,Cc1cccc(CC(=O)NC2CC(O)CN(C(=O)CN3CCC(C)CC3)C2)c1C 25957,N1(C(c2n(C)ccn2)=O)CC2(CC(NC(C3(C(F)F)CC3)=O)CO2)C1 25958,CC1CCc2sc(C(N3CCC(CNC(c4csc(Cl)c4)=O)C3)=O)cc2C1 25959,c1(C(N2CCC3C(CCN3C(C3C=CCN3)=O)C2)=O)c(Cl)ccc2c1OCO2 25960,c1(CNC2CCC(C(=O)NCc3cn[nH]c3)C2)ccccc1C(F)(F)F 25961,C(CC(C)(C)C)(C(=O)NCCC1CCCN1C(c1cc(C)nn1C)=O)OC 25962,c1(NC(C2CCN(C(C3CCCO3)=O)C2)=O)ccccc1NCC1CC1 25963,C(C(C)(F)C(C)(C)F)NC(CCCN(C(c1n(CC)c(O)nc1)=O)C)=O 25964,C1(CC=C)(N(C(=O)Cc2cocn2)CC)CC2CCC(C1)N2C(=O)CCC 25965,N1(Cc2nc(C#C)sc2)CCCN(C(=O)Cc2ccccc2)CC1 25966,N(C1CN(C(c2cncn2C2CC2)=O)Cc2ccccc21)C(CSCC(C)C)=O 25967,C(=O)(C(C(C)(C)C)NC(C1CN(C(c2ccc(C)c(F)c2)=O)CC1(F)F)=O)NC 25968,C(C(C)(C)C(=O)N1CC(C(N)=O)(CNC(c2nnn(C)c2C(F)F)=O)C1)SC 25969,c1(OC)cncc(C=CC(=O)NC2(CN(C(=O)CN3CCCC3C)C)CC2)c1 25970,Cc1cc(C(=O)NC2CCCC2NC(c2ccnc(O)c2)=O)nc(O)n1 25971,c1(C(N2CCC(SC)C2)C(=O)NCC(=C)C)ccc(Oc2ccccc2)nc1 25972,c1(CN2CCC(F)(C(=O)NC(CCC)C)C2)cc(C(=O)OC)ccc1OC 25973,c1(C(N2CC(C(=O)Nc3cc(Br)cc(Br)c3)C(O)CC2)=O)cccc2c1CCC2 25974,CCC(CCC(=O)NCC(CC(=O)NCC(C)(CC)CO)C1CCC1)OC 25975,C1(NC(C(c2n(C)ccc2)=O)=O)CCCN(CC(=O)Nc2ccsc2C(N)=O)C1 25976,C(C1=CCN(C(C2CCC(F)CC2)=O)CC1)NC(C(C)C1CCC1)=O 25977,C(=O)(CCCCCCCCC1CC1)NCC(CC)(C)NC(c1ccccc1C)=O 25978,c1(OC)cc(OC)c2c(c1)CCN(C(=O)C(C)Sc1cc(Cl)cc(Cl)c1)C2(C)C 25979,c1(C(=O)NC2CN(C(=O)NC3(COC)CC3)CC2C(F)(F)F)ncc(N)cc1Cl 25980,CCCCCCCCCCCCN(C(=O)CC1CCN1C(=O)OC(C)(C)C)C 25981,c1(C(N2C(C)(CNC(C3(C)C(C)CCC3)=O)CCC2)=O)cn2c(n1)CCCC2 25982,CC(C)(C(=O)NCc1cc(C(=O)NC2CN(C3CCC3)C2)on1)C(N)=O 25983,CC1(C)CC(C)(C)CC(O)(CNC(=O)CNC(c2cscc2Br)=O)C1 25984,C1(CNC(Cc2nc(C(C)C)sc2)=O)CN(C(=O)C=CS(C)=O)CC(C)(C)O1 25985,c1(C(=O)NCCCOCCC(=O)NCCc2nncs2)cccc(=O)o1 25986,C1(C(=O)NCC(CCOC)NC(C2COCCC2(F)F)=O)CC2(C1)OCCO2 25987,c1(C(N2CCC(N(C(=O)CCc3cccnc3C)CC)C2)=O)cc(C)ccc1N 25988,C12(CNC(CCc3ncn(C)c3)=O)CCC(NC(=O)COC3CCC3)(CO1)C2 25989,C1(NC(Cc2c(C)ncs2)=O)C2CC3C(C2)C13C(=O)NCCC1CC=CCC1 25990,c1(C(N2C(C)C(NC(=O)C(N)=O)CCC2)=O)cc2c(nc1O)CCC(C(C)C)C2 25991,CCC(C)(C(=O)N1CCC(C)N(C(=O)CCc2cc(C)no2)CC1)C(F)F 25992,C(=O)(CS(=O)(=O)CC(=O)NCC1CCN1C(=O)Cn1nc(C)nc1C)OC 25993,C(C(C)(C)C#CC(=O)N1CC(O)(C(F)(F)F)C1)NC(C(CC#C)C1CC1)=O 25994,CC1(C)CN(C(=O)C=Cc2cn[nH]c2)CC(CNC(=O)C(F)(F)CC2CC2)O1 25995,N1(C(CC2(C)CCOCC2)=O)CC2CC(NC(=O)CCN3CCOCC3)C(C2)C1 25996,Cn1cnc2c(NCc3ccn(C4CC4)n3)[nH]c(=NC3CCC=CCCC3)nc12 25997,Cc1ccc(F)cc1NC(=O)CC1(C)CN(Cc2ccc(Cl)cc2Br)C1 25998,C(=O)(C(=O)N=c1cc(C)o[nH]1)NCC1C(F)(F)CCN(C(CSCC)=O)C1 25999,c1(C(=O)NCCC(CCC)C)cc(C(N)=O)cc([N+](=O)[O-])c1 26000,Cc1nn2ccccc2c1C(=O)NC(CNC(C1CC1C(N)=O)=O)CC(F)(F)F 26001,N1(C(c2cc(OC)ns2)=O)CC(NC(=O)Cn2cnc(C#N)n2)C2CCCC2C1 26002,C(=O)(C(CNC(=O)Cc1coc(C)n1)CC1CCCC1)NCCCCOCC 26003,N1(C(c2ccc(N)c(O)c2)=O)CC(NC(c2cc(Cl)c(Cl)s2)=O)CC12CCC2 26004,c1(OC)ccccc1C(CNC(=O)Cc1ccc(F)cc1)NC(=O)CO 26005,C12(NC(c3cc(NC)nc(Cl)c3)=O)CCCC1CN(C(=O)Cn1ccc(C)n1)C2 26006,Cc1nc(NC2CCC3CN(C(C4(CO)COC4)=O)CC23)ncc1[N+](=O)[O-] 26007,C1(C(C)(C)O)(CNC(c2ccnn2CC(F)F)=O)CN(C(c2ccccc2)=O)C1 26008,c1(C(N(C)CC2CC(F)CN2C(=O)C(F)=C2CCCC2)=O)cc(N)ccc1O 26009,c1(CCC(=O)NC2(C)CC(NC(C3C(C)OCC3)=O)C2)ccc(C#N)cc1 26010,c1(C(CC(=O)NC2CC(F)(CNC(c3c(SC)ccs3)=O)C2)O)ccc(F)cc1 26011,C1(C(N2CC(N(C(=O)CC3CCC3)C)C2)=O)CCCCC1C1CC1 26012,c1(CC(=O)NC(CNC(COCCOCC)=O)(C)C2CCC2)coc(C(F)F)n1 26013,C1(C(N(CC(=C)C)CC)=O)CCN(C(c2cnn(C)c2Cl)=O)C1(C)C 26014,CC(C)S(=O)(=O)C1CCN(C(CCCCC#N)c2nnnn2CCCSC)CC1 26015,C1(CCNC(=O)COC2CCOCC2)CSCCN1C(C1CCC(F)(F)C1)=O 26016,C1(NC(C2(C#C)CCN(C(c3cc(CC)nn3C)=O)C2)=O)CC2C(O)C(O)CC12 26017,c1(C(=O)NC(CC)C(=O)NC2COC3(CCC3)C2)coc2c1COC2 26018,c1(C(C(=O)NCC(C)(C)OCCNC(Cc2ccc(C)o2)=O)C)cccc(F)c1 26019,N1(C(C(C)CC(N)=O)=O)CCC2(CCN(C(c3ccc4nc[nH]c4c3)=O)C2)C1 26020,N1(C(c2scc(CNC(C3CN(C)C3)=O)c2)=O)CCCC2CC12.OC 26021,N1(C(c2c(OC)cccn2)=O)CCC2CN(C(c3ccnc(C)c3N)=O)C(C)C12 26022,C(C)(C(=O)NOC(C)C(=O)OC)NC(c1c(CCC)[nH]cc1)=O 26023,C=CCCCCCCCC(=O)NC(C)CN(C(c1nccn1C)=O)CC 26024,c1(C(N2CCC3CN(C(C(F)=CCC)=O)C3C2)=O)n[nH]c2c1CC(C)OC2C 26025,C1(NC(C(C(C)C)N(C)C)=O)CN(C(=O)C=CBr)CC1C1CC1 26026,C(=O)(C(C)(C)C(F)F)NC(C(C(C)C)Nc1ncc(F)cn1)C 26027,c1(NCC2CCN(C(C)C)C2)cc(=NCc2ccc(-n3ccnn3)cc2)[nH]cn1 26028,C1(C#N)(C(N2CCC(CC(=O)NC3(C)CCCC3)C2)=O)CC(F)(F)C1 26029,c1(CCNC(C(C)OCC)=O)cnn(C)c1C1CN(C(=O)COCCOCC)C1 26030,c1(NC(c2scc(-c3cc(C(=O)NC)ncc3)c2)=O)ccc2cnn(C)c2c1 26031,C12(NC(c3cc4c(O)nnn4cn3)=O)CC(CO)(C1)OC21COC1 26032,N1(C(C(C)(C)NS(C)(=O)=O)=O)CC2(C1)SCCC2N=c1[nH]ccnc1F 26033,c1(C(=O)NCCC(C)N(C(C2C(C=C)C2)=O)C)cc(F)cc2nn[nH]c12 26034,C(C1=NOC2CN(C(=O)CC3CC3)CC12)NC(c1cc(CC)c(C)cc1)=O 26035,C=CC(CC(=O)NCCCCNC(C1CC1OCC)=O)c1ccccc1 26036,N1(C(C(CN(C)C)(C)C)=O)CCC(C2CC2)(CNC(=O)CCCC2CCCO2)C1 26037,c1(C(C(C)(C)C)N(C)C)nc(-c2cncnc2)nn1-c1ccccc1 26038,C1(NC(c2cnc(C3(C)CC3)o2)=O)CCCN(C(c2coc(Br)n2)=O)CC1F 26039,Cc1nc(NC(C2CCCN2Cc2ccncc2O)=O)cnc1Cl 26040,C1(NC(C(CC)N(CC)CC)=O)CCN(C(=O)CC(F)(F)F)CC(O)C1 26041,N1(C(C(CCNC(C(CC)NC(C)=O)=O)O)=O)CC(O)CC12CCOC2 26042,N1(C(C2(C)CCN(C(c3ccc(C#N)[nH]3)=O)C2)=O)CC2CC1CC2CF 26043,C1(NC(C(COC)(C)OC)=O)CN(C(=O)COC(C)=O)CC2(CC2)C1 26044,O=C(C#Cc1ccccc1F)NC1(c2nn[nH]n2)CC12CCCC2 26045,N1(C(c2ccc(CCC)[nH]2)=O)CC(NC(=O)CCS(N)(=O)=O)CC12CCOCC2 26046,c1(CC(=O)N(C)CC2CCN(C(c3ccon3)=O)C2)ccc2c(n1)OCCO2 26047,c1(N2CC(C)C=C(C)C2)nc(NCCc2c[nH]nc2C2CC2)c2ccsc2n1 26048,C(=O)(CC(CC1CC1)NC(=O)C(C)OCC1CC1)N1C(C=C)CC1 26049,N12CC(C3(CC3)C1)CC(=O)N(CC#C)CC2=O.C1(C(=O)OC)CCOC(C)C1 26050,C(CN=c1[nH]c(=NC2CC2C(C)(C)C)c2ccccc2[nH]1)c1c(C)nc(C)s1 26051,N1(C(c2c(CNC(=O)CC3CCCC3)c[nH]n2)=O)CC=C(CO)CC1 26052,C1(CC)C(NC(c2cc(O)nc(Cl)c2)=O)CCCN1C(=O)CCS(N)(=O)=O 26053,c1(NCC(CCC)(F)F)ccc(Cl)cc1N1CCOCC1 26054,CN1CCCCC(C(N2CC=CC(NC(c3csc(C(C)(C)C)c3)=O)C2)=O)C1=O 26055,CCCC(CC)C(=O)NCCCN1CCC(NC(=O)C(C)C(=O)OC)C1 26056,CCC(C)C(=O)NNC(=O)Nc1ccc2c(C)nnn2c1 26057,N1(C(C2C(CC)OCC2)=O)CC(OC)C(NC(=O)CC23CCCC2C3)C1 26058,c1(CC(C(=O)NCCC(C)N(C)C(c2ocnc2C2CC2)=O)O)ccccc1Cl 26059,N1(C(C(C)Sc2ccccn2)=O)CC2CCC1C(C(=O)NCC1CCCC1O)C2 26060,C=CC1CCCN1C(C1(CC)CCN(C(=O)CCOCCCC)C1)=O 26061,c1(C(=O)NC(CC)CNC(=O)CC(C)SC)ccc2c(c1)COC2=O 26062,N1(C(CNC(=O)Nc2ccccc2)=O)CC2C(NC(C3(O)CCCCC3)=O)C2C1 26063,c1(OCC(C(=O)OC(C)C)(C)O)cc(C(N)=O)ncc1Br 26064,c1(CC(N2C(CNC(c3c(C)nco3)=O)CCCC2)=O)cc2ccccc2s1 26065,Cc1ccc(C(N2CCOCC2CC(=O)NCC2COCCO2)=O)nc1O 26066,c1(CC(N2C3C(NC(C4CC(C)SCC4)=O)C(C3)C2)=O)ccccc1[N+](=O)[O-] 26067,C(=O)(C(CC(C)C)ONC(C1CC2(CC(=O)C2)C1)=O)NC(CC)C1CCC1 26068,C1(NC(=O)CN2CC(CNC(=O)Cc3ccns3)C2)CCCCN1C1CCCC1 26069,[N-]=[N+]=NC1CCCCC1C(=O)NCC1CC(F)(F)CN1C(=O)CC1C=CCC1 26070,CCCCCC(O)CC(=O)NCC1(O)CCCN(C(=O)C2=CCCC2(C)C)CC1 26071,C1(C(=O)NCCC2CN(C(=O)CC(C3CCC3)C3CCC3)C2)(COC)C=CCC1 26072,c1(N(C2CC3(CNC3)C2)C(c2ccc(OCC)cc2)=O)ccc(O)cc1 26073,c1(N(CC(C)C(C)(C)C)C)nc(N2CCCC(C)(F)C2)nc2ccc(Cl)cc12 26074,C1(C(N2CC(CCCCC)C2)=O)CCCC(NC(C2(F)CC=CCC2)=O)CC1 26075,c1(CC)ccc(F)cc1NC(=O)CCN(C(C12CCC(C1)C2)=O)CC1CC1 26076,CN1CC2CCC(C1)N2C(C1CCC(O)CN1C(=O)C1=C(Cl)CCOC1)=O 26077,CC1=C(C(=O)N2CCC(NC(c3cnn(C(C)C)c3Cl)=O)C(C)(C)C2)CCCO1 26078,N1(C(Cn2c(C)cc(C)n2)=O)CCOC2CN(C(c3cccnc3)=O)CC12 26079,c1(CC(=O)NCC(CC)(C)NC(c2ncoc2C)=O)cc(Br)ccc1F 26080,c1(C(=O)NCC(CCOC)NC(=O)CC2CCC(C)(C)C2)[nH]c(C2CC2)nc1C 26081,C(=O)(CC(C)(C)CC)N1CCC(N(C(C2(NC(C)=O)CCCCC2)=O)CCO)C1 26082,c1(C(N2CCC(F)(CNC(c3c(CC)cccc3)=O)C2)=O)ncc(N)cc1Cl 26083,N1(C(c2ncc(C)nc2)=O)CCCC(NC(C2(C(C)C)CNC(=O)C2)=O)CC1 26084,C1(CNC(C(C)NC(N)=O)=O)(CO)CCN(C(=O)C=CCF)CC1 26085,Cc1cc(C2CCN(S(=O)(=O)CCC(O)COc3ccccc3C)C2)cc(C)c1 26086,N12CCOCC13CN(C3)C(=O)C2c1occ(C)c1.C(C)(C)(C)OC(C)=O 26087,c1(N(C(CN(C)Cc2ccc(C)c(C)c2)=O)C2CCC2)c(Br)cccc1[N+](=O)[O-] 26088,N1(c2c(Br)cnc(C)n2)CCN(C(=O)CCc2ccccc2Br)C(C#N)C1 26089,c1(OC)cc(C(=O)OC2CCCN(C(N3CCCCC3=O)=O)C2)cc(Br)c1 26090,N1(C(c2cncc(C)c2Cl)=O)CCCC(C2CC2NC(C2(N(C)C)CCC2)=O)C1 26091,N1(C(c2cc(COC)on2)=O)C2CCC1CC(N(C)C(c1cnc(SC)s1)=O)C2 26092,N1(C(Cn2cc(CNC(C3(C)CCNC3=O)=O)nn2)=O)CC(O)C(C2CC2)C1 26093,N1(C(CCC#C)=O)CC2(CCCCN(C(=O)C(C)C3CCCO3)C2)C1 26094,N1(C(c2c(CC)occ2C)=O)CCCCC(NC(=O)C(C(C)(C)C)N(C)C)C1 26095,Cc1cnc(C=CC(=O)NC2COCC2NC(=O)CC2COCC2O)[nH]1 26096,c1(OC)cc(C)ccc1C(=O)NC(C1CCN(C(=O)CC=CC(C)(C)C)C1)(C)C 26097,N1(C(CC2C(OC)CC2)=O)CCN(C(c2cocn2)=O)C(c2ncc[nH]2)C1 26098,C1(CNC(C2(C(C)C)CC2)=O)CCC2(CN(C(=O)Cn3ccnn3)C2)O1 26099,C(=O)(C1CCc2c[nH]nc21)NC1(C(=O)NC(C2CCCCC2)C)CSC1 26100,N1(C(CCC#CC)=O)CCCC(C(=O)N(C)CC2CCOC2)CC1 26101,c1(C(=O)NCCC2N(C(C(CO)N(C)C)=O)CCCC2)cc(S(N)(=O)=O)cn1C 26102,Cc1[nH]nc(C(=O)NCC2CCCN(C(C3CC3C)=O)C2)c1C 26103,C1(CC)CN(C(=O)C(C)CN2CCCCC2)CCN1C(=O)C(C)C 26104,c1(C(=O)NCCCCN(C)C(C2CC2c2cccs2)=O)c[nH]nc1C(C)(F)F 26105,N1(C(Cc2cnc(C)o2)=O)CCCC2(NC(=O)CSc3nccn3C)CC2C1 26106,c1(C(N2CCN(C(c3cnn(C(C)C)c3N)=O)C(C)C2)=O)nc[nH]c2ncnc1-2 26107,N1(C(Cn2c(N)cc(C)n2)=O)CCCC(N(C)C(c2ccccc2O)=O)CC1 26108,c1(CC(=O)NCCOCCNC(COCCCCC)=O)ccc(F)c(Cl)c1 26109,c1(-c2ccc(CCC)cc2C)ccc2oc(C(=O)NC(CC)C(F)(F)F)cc2c1 26110,c1(C(=O)NC)noc(CNC(c2cscc2C)c2nnnn2CCCF)n1 26111,c1(NC(c2c(OC)cncc2)C)ccc(S(=O)(=O)NCC2C3CCCOC23)cn1 26112,c1(CC)[nH]nc(C(=O)NC(CN(C(=O)C(C)(F)F)C)CC)c1Cl 26113,N1(C(c2c(C)oc(Cl)n2)=O)CCN(C(=O)CN2CCSCC2)CC1C1CC1 26114,C1(CNC(C2N(C=O)CCC2)=O)CCCN(C(c2cnc(C(F)F)nc2)=O)CC1 26115,c1(C(N2CCC(=CCNC(C(C(C)C)C)=O)CC2)=O)c(F)ccc2occc12 26116,O=S(=O)(c1ccc(N2CC3CC3(CO)C2)cc1Br)NCc1cn2ccccc2n1 26117,Cc1ncc(S(N)(=O)=O)cc1C(=O)NC1CCCCN(C(=O)CC2CCC2)C1 26118,C1(CC)CN(C(=O)CN2CC(C)(OC)C2)CCN1C(=O)CN(C)C 26119,c1(C(N2CC(C(=O)NCc3cc(C)on3)OCC2)=O)cc(Cl)cnc1Cl 26120,C#CCC(C)(C(=O)N1CCC(CN(C)C)C1(C)C)NC(c1ccc(F)c(C)c1)=O 26121,C(=O)(C1=COCCO1)NC1C(CNC(c2cc(C(C)=O)cn2C)=O)C1 26122,N1(C(CCOC)=O)CCC(C(C)NC(=O)CC2CC3CC3C2)CC1 26123,C1(NC(C(Cc2cccc(Br)n2)N(C(CC(C)O)=O)C)=O)(CO)CCOCC1 26124,c1(OC)c(F)ccc(F)c1CN1CCC(C(=O)NC(c2ccc(Cl)cc2)C)C1 26125,C12OC3(C)CC1(C3)CNC2=O.c1(NC(=O)OC(C)(C)C)ccccc1CC1CC1 26126,c1(N2CCCC(NC(c3c(C)nn[nH]3)=O)C2)ccc(Cl)cc1[N+](=O)[O-] 26127,C1(OC)COCCC1N(C(C1CCCOC1)C(=O)NC1CC1)C 26128,c1(C(=O)NC2C(NC(CSC(C)(C)C)=O)CS(=O)(=O)C2)ccc2nncn2c1 26129,N1(C(C2CC(N(C(C(C)NC(CC)=O)=O)C)C2)=O)CCC(CO)C1(C)C 26130,C1(CN(C)C(c2ccc(F)s2)=O)CCN(C(C2(O)CCC2)=O)C1 26131,S(=O)(=O)(c1ccc2[nH]c(=NCc3ccsc3)ccc2c1)NCCCCN(C)C 26132,C(=O)(CP(C)(C)=O)NCC(CN(C(=O)C(C)O)CC)(C)C 26133,CCCCCCC(CC)C(=O)NCC1COCCN(c2nccn3nnnc23)C1 26134,C(N=c1[nH]c(=NC(CCO)c2ccccc2F)[nH]c2ccccc12)C1(C)CCC1 26135,C1(C(C)NCCNC(c2ccc(Cl)o2)c2nnnn2C2(C)CC2)CCC(F)(F)CC1 26136,N1(C(c2ccon2)=O)CCC2C(CCCN2C(=O)Cc2cnc(C(F)(F)F)s2)C1 26137,C(=O)(C1CCCc2ncc(C)n21)N1C(CNC(c2c(OC)ccc(OC)n2)=O)CC1 26138,CCS(=O)CC(=O)NCC(=O)NCC(=O)NC(c1nccs1)CC 26139,CCC(C)C(C)(O)CNC(C1CC(C)CN(C(=O)Cc2ccc[nH]2)C1)=O 26140,c1(SC)nc(=NCC2(NC(C3CC3(C)Br)=O)COC2)s[nH]1 26141,CCCCCCCCC(=O)NC(C)CN(C(=O)Cn1cc(F)ccc1=O)CC 26142,C1(NC(C(=O)NC(C)C)=O)CCC(F)(CNC(c2csc(Cl)c2)=O)C1 26143,C1(C(=O)NC2CC3(CN(C(Cc4c(C)non4)=O)C3)C2)CCCC1S(C)(=O)=O 26144,C1(CC(=O)N(C(C)C(C)(C)O)C)N(C(c2ccncc2Cl)=O)CCC1(C)C 26145,c1(OCCC(=O)NCCC2CCCN(C(=O)Cc3ccsn3)C2)ccc(Cl)cc1 26146,C1(C(=O)NCC2N(C(CC3CN(C)C3)=O)CC(F)C2)CC1C1CCCC1 26147,N1(C(c2cncc(C)c2C)=O)CC2CC(NC(=O)C(C)(C)CC(C)C)CC2C1 26148,N1(C(C(C)CO)=O)CCCCC1CCC(N1CCC(C(N)=O)C1)=O 26149,C(=O)(CC1=NN(C)C(=O)C1)NCC=CCNC(c1cc(OC)n(C)n1)=O 26150,N1(CC)CCC(n2nc(-c3cncc(F)c3)nc2COC)CC1 26151,C1(N(C(COC(C)=O)=O)C)CCCC(NC(=O)Cc2cnn(C)c2C)C1 26152,C1(CNC(C2CCN(CC(C)C)C2)=O)CC(C(=O)N(CCC#N)C(C)C)=NO1 26153,C1(CC(=O)NC2CC2NC(c2cncc(CO)c2)=O)CN2CCN1CC2 26154,C1(NC(=O)NC2(O)CN3CCC2CC3)CC2CC(NC3C4CC5C(C4)C35)C1C2 26155,[N-]=[N+]=NC1(C(=O)NCC(O)CF)CCN(C(=O)CC2CCOC2=O)C1 26156,S(=O)(=O)(CCC(F)(F)F)N(C1CN(C(C2CC2(F)F)=O)CC1O)C 26157,c1(NC(N2CCC(C)(c3ccccc3)C2)=O)c(I)cc(F)c(Br)c1F 26158,C1(OC)(OC)CCC(CN(C(C(C)C)c2cnn[nH]2)C(C2CCC2)=O)C1 26159,N1(C(CC2(C)CCN2C(=O)CC2CC(F)(F)C2)=O)CCOC(C)(CO)C1 26160,C1(C(=O)NCc2cn(CC=C)nn2)C2CCC(C2)C1NC(C1CCC(NC)C1)=O 26161,N1(C(Cc2cc(CC)nn2C)=O)CC2CC(NC(c3cc4scnc4[nH]3)=O)C1C2 26162,N1(C(c2c(NC(C3(CC)CCCC3O)=O)n[nH]c2)=O)CCNC(=O)C1CCO 26163,C1(NC(COC2C(C)CCCC2)=O)CCN(C(=O)CS(C)(=O)=O)CC1O 26164,C1(NC(C(CC)C)=O)CCC2(CC1)CN(C(c1cscc1Cl)=O)CCO2 26165,C(CC(C)N(C(=O)CCSC1CCCC1)C)NC(C1C(CN(C)C)C1)=O 26166,C(CC(C(=O)NOCC1(C)CCC1)NC(C1CC2(CCCO2)C1)=O)=CC 26167,c1(C(N(CCCNC(=O)CN2CCOCC2=O)C(C)C)=O)cc2ccsc2n1C 26168,c1(C(C)N(C2CS(=O)(=O)C2)C(=O)C2CC2)cccc(F)c1 26169,CC(N=c1cc(C(F)(F)F)nc(Cl)[nH]1)C(c1ccccc1)NC(=O)C(C)O 26170,C1(NC(c2c(C)nc(CCC)s2)=O)CC2(CCN(C(=O)CCOC(C)C)C2)C1 26171,Cc1cccc(C(=O)NCC2(CNC(=O)C=CC3CCC3)CCCC2)c1[N+](=O)[O-] 26172,N1(C(C2N(C(C)=O)CC(O)C2)=O)CCN(C(=O)C(F)(F)C(C)O)CC1CO 26173,c1(C(=O)NC23C(CN(C(CNC(C(C)CO)=O)=O)C2)C3)ccc2c(c1)CCCC2 26174,C1(NC(CC2CC(=C)C2)=O)CCCCC1CNC(=O)CCC1(O)CCC1 26175,Cc1ccc(CC(=O)NC(CNC(C2CC(n3ccnc3)C2)=O)C2CC2)cc1C 26176,c1(CC(=O)NCC(C)CN(C(=O)Cc2cnns2)C)cccc(OC(F)(F)F)c1 26177,C1(C(=O)OC)CC(OC)CN(C(=O)C(C)Oc2ccccc2)C1.C1(=O)CO1 26178,CCC(C)CCC(=O)NCCOC1CN(C(=O)CCCc2ccc(C)s2)C1 26179,c1(C(N2C(CCNC(C3CCO3)=O)CCC2)=O)csc2ccc(F)cc12 26180,N1(C(c2c[nH]c(=NC)s2)=O)CC(NC(=O)C(Br)=C(C)C)CC(C)(C)C1 26181,c1(C(=O)NCC2C3N(C(C4CC(OC)C4)=O)C(CC3)C2)c(Cl)c([N+](=O)[O-])nn1C 26182,CCC(CCC(=O)N(CC(C1CCC1)OC)C)NC(c1ccc(F)c(O)c1)=O 26183,C1(C)(CNC(C2C(CNC(c3cc(COC)no3)=O)C2)=O)CNC(=O)O1 26184,C1(CC=C)(NC(=O)C(O)C2CC2)CCN(C(c2sc(Br)cc2C)=O)C1 26185,c1(SC)c(C(=O)NCC2CC3(CC3)CN2C(c2cnn(C)c2)=O)cccc1F 26186,c1(NC(c2cc(C)c(Cl)cc2Cl)=O)cccc2oc(C(=O)O)nc12 26187,CCCCCC(=O)NCC(C1(O)CN(C(c2ncn(C)n2)=O)C1)(C)C 26188,c1(N2CCC(C(C)NC(C(C)Oc3cccnc3)=O)C2)nc(Cl)c(C#N)s1 26189,C1(C(=O)NCCCc2n(C)nnn2)CCN(C(c2ccc(=O)n(C)c2)=O)C1(C)C 26190,C1(N(C(CC2CN(C(C(C)n3cccn3)=O)C2)=O)C)CCN(C2CC2)C1 26191,C1(CC(=O)NCC2CCCO2)CCN(C(C2CCCC2)=O)C1.C1C(=O)N1 26192,c1(CNC(=NCC)NCC23COCC2C3(F)F)ccc(OC(C)(C)C)nc1OC 26193,NS(=O)(=O)CCC(=O)NCCC1(CNC(=O)CC2CCC(O)C2)CC1 26194,C1(C)(CNC(COCC(=C)C)=O)CCC(NC(c2ccn(CC)c(=O)c2)=O)CC1 26195,c1(CCCC(=O)NCCC(C)NC(C2COCCO2)=O)ccc(F)c(F)c1 26196,CC1CCN(C(C2(N=[N+]=[N-])CCN(C(c3ccn(C(F)F)n3)=O)C2)=O)CC1O 26197,C(C1CN(C(c2coc(C(F)F)c2)=O)CC1C(=O)NC1(CO)CCCC1)=CC 26198,CCCCC(CC)C(=O)NC1CN(C(c2cccc(C(N)=O)n2)=O)CC12CC2 26199,C(=O)(C(C(C)(C)C)n1cc(C2CN(C(c3cnn(C(C)C)n3)=O)C2)nn1)OCC 26200,C(=O)(CS(=O)(=O)C1CC1)NCC1(C)CCN(C(C2CCCC2C(F)(F)F)=O)C1 26201,c1(OC)ccc(C(=O)N(CCC(C)NC(C2(C)CC2(C)C)=O)C)cc1S(N)(=O)=O 26202,N1(C(c2c(Cl)ccc(C#C)c2)=O)CC2(C1)C(NC(=O)C=CC(C)C)CCS2(=O)=O 26203,Cc1nc2c(NC(C3C=CC(NC(c4cc(F)cnc4Cl)=O)C3)=O)cccn2n1 26204,N1(C(=O)CN2CCOCC2)CC(C2CCCCN(C(=O)C(F)(F)CO)C2)C1 26205,CON1CCC(C(N2CCCC2CC(=O)NC(C)CN(C)C(C)C)=O)CC1 26206,C1(C(=O)NC2CN(CCCCC)C2)C=CC(NC(=O)CC(Cl)Cl)C1 26207,c1(OC)cc(OC)cc(C(C(=O)O)NC(c2ncoc2C(C)(C)C)=O)c1 26208,CC1CCC(CNC(=O)COCC2CCCO2)CN1C(=O)C=Cc1nccs1 26209,Cc1sc(Cl)c(C(N2CCCC(C)(NC(=O)CCNC(C3CCC3)=O)C2)=O)c1C 26210,N1(C(c2cc(C)cc(O)c2)=O)CCN(CCOCC(F)(F)F)CC(C)(F)C1 26211,C1(CCNC(C2C(CN(C)C)C2)=O)CN(C(c2cc(N)ccc2O)=O)CCCO1 26212,C(=O)(CC1=NNC(=O)C1)N1C(CCOC)CN(C(c2ccncc2OC)=O)CC1 26213,c1(C(N2CC(NC(C)=O)CC(C)(C)C2)=O)nnn2cc(C)nc(O)c12 26214,N=c1ncc(C(=O)NCC2(C(F)F)CCN(C(=O)Cc3ccc(F)cc3)C2)c[nH]1 26215,C(CNC(C)=O)(C(C)C(C)C)NC(C1(OCC)CCOCC1)=O 26216,N1(C(C(CC)C(F)(F)F)=O)CC2(C=C(C(=O)NCC3CCSC3)CO2)C1 26217,Cc1cc(C)n(CCCCNC(=O)CC2CCN(C(c3ccco3)=O)C2)n1 26218,C(C#N)(C(=O)C(C)(C)CNC(c1ccc(C)cc1)=O)c1ccc(OC)cc1 26219,c1(OC)cc(C(=O)NC2CN(C(C3CCC4CC34)=O)CC2F)sc1Br 26220,N1(C(C=CC(CC)=CC)=O)CC(O)(C2(CNC(c3ccc(=NC)[nH]c3)=O)CC2)C1 26221,Cc1nsc(C(N2CC(F)(C(=O)NCCN3C(=O)CCC3=O)C2)=O)c1N 26222,N1(C(C2C(C=C)C2)=O)CC(CNC(=O)C(=O)N(C)C)(COC)C1 26223,c1(N2CC(OCC)(CNC(=O)CC(O)c3ccccc3)C2)ccnc(CO)n1 26224,S(=O)(=O)(c1cn(C)nn1)NC(=O)Nc1cccc(C)c1OCc1cccc(Cl)c1 26225,c1(C(=O)NCC(C)N(C(=O)COc2ccc(F)cn2)C)cnc(Cl)cn1 26226,C(Cn1ccnn1)(C(=O)NCCc1nc(O)n[nH]1)NC(C1C(C)(C)C1)=O 26227,c1(C(=O)NC2CCN(C(C(CC=CC)C)=O)CC2F)ccc2nccc(C)c2c1 26228,c1(C(c2n(CCSC)nnn2)NC2C3CCC2CC3)cc(Cl)ccc1Br 26229,C1(NC(C(C)(C)SC)=O)CC2CN(C(C3CC3(F)F)=O)CC12 26230,C(CC(C(=O)N1CCC(C)(C(N)=O)C1)NC(c1cccc[n+]1[O-])=O)N(C)C 26231,c1(C(N2C(CC)C(C(=O)N(C3CC3C3CC3)C)CC2)=O)cccc(C)c1N 26232,C1(CCC)CN(C(=O)Cc2csc(Cl)n2)CCN1C(=O)C(C)OCC 26233,N=c1[nH]c(CCC(=O)NCCOC2CN(C(C3CC3Cl)=O)C2)cs1 26234,Cc1cc(CCNC(=O)CCn2cc(CC(C)O)nn2)ccn1 26235,C1(C(=O)NC(c2ncc[nH]2)CC)C=CCN(C(=O)CN2CCCCC2)C1 26236,CCCC(C(=O)NC(C)C(=O)NCC(C)(CC)CC)NC(N)=O 26237,N1(c2nc(C)c(F)cn2)CCc2ccc(NC(=O)CC3COCCO3)cc2C1 26238,n1(CC(=O)NC2C(NC(c3c(C)ncn3O)=O)CCCC2)ccc2ccccc12 26239,c1(C(=O)NCC(=O)N(CCNC(C2CCCC(=O)O2)=O)CC)cc(F)cc(F)c1 26240,N1(C(C2C(C)(C)CCC2)=O)CC(NC(=O)CCc2cccc(F)c2F)C(C)(C)C1 26241,C1(CCNC(C(C)(C)SC)=O)CN(C(=O)Cc2nnc(O)s2)CC(C)O1 26242,c1(CC(=O)NC(C2CC=CCC2)C(=O)NCCN(C(=O)OC)C)ccccn1 26243,CC(CC(N)=O)C(=O)NC1CC(CNC(c2cc(C3CCOCC3)nn2C)=O)C1 26244,N1(C(c2n(CC#C)ccc2)=O)CC2CCC2(CC(=O)N(CC)CC)C1 26245,c1(CC(=O)NCC2(NC(c3cccc(F)c3O)=O)COC2)nc2ncccn2n1 26246,N1(C(C(C)NC(=O)OC)=O)CC(CCNC(=O)C(C)N2CCCC2)OC(C)C1 26247,Cc1cc2c(cc1C)C(C(=O)N1CCCC1CNC(c1cnc(S)[nH]1)=O)CO2 26248,N1(C(C(C)=CC2CC2)=O)CCN(C(C2(NC(C)C)CC2)=O)CC1CS(C)(=O)=O 26249,Cc1cccc(C)c1CCC(=O)NC1CC12CC(NC(=O)CC13CCCC1C3)C2 26250,CCC(C)C(O)C(=O)NC1CCN(CCNC(=O)C(F)(F)C2CCCC2)CC1 26251,CC1(C)CC2(CC(C(N3CCN(C(c4ccccc4Cl)=O)CC(CO)C3)=O)C2)C1 26252,CC(C)C(CNC(c1ccncc1N)=O)C(=O)N1CCCC(F)(F)C1 26253,c1(C(N2CC3C(CNC(C(C)=CC)=O)(C3)C2)=O)cccc2cccc(Cl)c12 26254,c1(C(N2CCC(c3cccc(C#N)c3)C2)=O)c(F)ccc2c1OCO2 26255,c1(NC(c2ccc(C(O)C3CC3)cc2)c2n(C)nnn2)ccccc1OC(F)F 26256,C=Cc1ccc(C(=O)NC(C)CN2CCN(C(=O)C(C)SCCOC)CC2)cc1 26257,C(=O)(CC(O)CC(C)(C)C)N(C(CC(=O)NC(CCC)C1CC1)C)C 26258,N1(C(CCOc2c(CC)cccc2)=O)CC(C2CN(C(=O)C(Cl)=CCl)C2)C1 26259,C1(NC(C2(C)CC(=C)C2)=O)CCC(F)(CNC(=O)COCC2CCCCO2)C1 26260,CC(C)C(F)(F)CC(=O)N1CCCC(N(C(=O)C(c2ccc(Cl)cc2)C)C)C1 26261,c1(OC)cc(C=CC(N2CC(F)CC2CNC(c2cnc(Cl)s2)=O)=O)ccc1N 26262,Cc1cc(C(=O)NC2CCN(C(=O)Cc3ccc(C)s3)CC2F)c2[nH]cnc2c1 26263,n1(CC)cnc2c(NCC(C)(C)OC)[nH]c(=NCC(C(C)(C)C)OCCO)nc12 26264,C1(C(N(CCCCN(C(c2ccc(COC)o2)=O)C)C)=O)CCCCCCC1 26265,c1(C(N2C(C(C)NC(C3(C)CS(=O)(=O)C3)=O)CCC2)=O)cn(C)c2ccccc12 26266,N1(C(C(CC)(C)O)=O)CCC2(CCCC(CNC(C3(C(C)C)CCC3)=O)O2)CC1 26267,c1(NC(C2N(C(COCC#C)=O)CC2C)=O)cncc([N+](=O)[O-])c1 26268,C1(CNC(C(CSC)C)=O)CCC2(CCN(C(=O)CC3CC=CC3)CC2)O1 26269,c1(C(N2CC(C(=O)OC)C(CC(C)(C)C)C2)=O)cnn2cc(Br)cc(OC)c12 26270,N1(C(c2n(C(CC)CC)ncc2)=O)CC2C(CNC(c3ccc(Br)o3)=O)C2C1 26271,c1(OC)cc(C)c(C(=O)NCC2(F)CCN(C(C3COC(=O)N3)=O)C2)cn1 26272,C1(NC(c2c(CC=C)cccc2)=O)CN(C(=O)C(O)C=CC)CC12CCC2 26273,C1(NC(c2c(C)nc(C(C)C)s2)=O)(CNC(=O)COC(F)(F)F)CCCCC1C 26274,C=CCC(CC=C)C(=O)N1CCC(C(=O)NC2(C)CCC(C)(C)CC2)CC1C 26275,Cn1nnc2c1CC(C(N1CCC(NC(=O)COCc3nc[nH]n3)C1)=O)CC2 26276,C1(C(N(C2CC(NC(C3(C(F)(F)F)CCC3)=O)C2)C)=O)CCCOC1 26277,c1(OC)ccc(C(=O)N(C(C)C(=O)Nc2cccc(Cl)c2)C2CC2)nn1 26278,c1(C(=O)NC(C)CNC(=O)C(C)Sc2ccccc2)ncc2ccccc2c1N 26279,c1(C(N)=O)nn(CC(C2CCC23CCNCC3)=O)c(=O)c2ccccc12 26280,C(=O)(C1=C(Cl)CCOC1)NCC(C1CCC1)NC(C1(C(=O)OC)CCCO1)=O 26281,N1(C(c2cnn(CC)c2)C(=O)NC(CC)C)CC(CC(=O)OC)C(O)C1 26282,C1(CCN(C(c2n(CC#C)ccc2)=O)C)CCCCN1C(=O)COCCOC 26283,c1(CNCCCCC(=C)C)cnn2ccc(OC)cc12 26284,CC1(C)CN(C(=O)CC2(CO)CCC2)CC1NC(c1ccccc1F)=O 26285,N1(C(c2ccc(Cl)cc2Br)=O)CCC2(CCN(S(=O)(=O)c3cccc(F)c3)C2)C1 26286,c1(OC)cc(F)cc(F)c1NC(=O)C(C)(C)C1CCCCC1 26287,c1(CNC(=O)NC2(C3CC[Si](C)(C)C3)CC2)cnn2ccsc12 26288,C(=O)(CCC(F)F)NC(C1(O)CN(C(c2cc(N3CCCCC3)ncn2)=O)C1)C 26289,C(C1CCOCC1)=CC(=O)NCC1CC(Cc2cn(C3C=CCCC3)nn2)CO1 26290,Cc1nc(=N)[nH]cc1C(N1CCC(N(C(=O)C(C)O)C)C1)=O 26291,c1(C(C(=O)NC2CCC(NC(C3C(C)(C(F)(F)F)C3)=O)C2)O)cccc(Cl)c1 26292,C1(CCNC(c2cccc(C)n2)=O)CCN(C(c2cnn(CCO)c2)=O)C(C)C1 26293,N1(C(C(CC(C)C)C(C)C)=O)CCc2cc(CNC(C3CC=CC3)=O)ccc2C1 26294,Cc1cc(NC(=O)COC(c2ccccc2N(C)C)=O)cc(C)c1N.C(=O)C1CC1 26295,N1(N(c2ccccc2)C)CC2(CC(NC(C3CC(C)(C)C3)=O)C2)C1.C1(C=O)(N)CC1 26296,N1(C(C(C=C)(C)O)=O)CC(C2CCCN(C(=O)C(c3ccccc3)F)C2)C1 26297,C1(C(=O)NC(CCOC)COC)CN(C(C2CC(C)=NO2)=O)CC1(C)C 26298,Cc1ncnc(C)c1C(=O)NCc1cc(C(=O)NCCC2CCCC2)cs1 26299,O=C1Cc2c(C(N3CC4(CC4)CC3CNC(=O)C(F)C3CCC3)=O)cccc2N1 26300,C1(NC(C(OCC)OCC)=O)CCN(C(=O)CC2CC(C(F)F)C2)CC1C(C)C 26301,c1(C(N(CCCNC(CC(CCC)C)=O)CC)=O)csc(=NC2CC2)[nH]1 26302,c1(C(C(=O)NCC(CN(C(c2csnn2)=O)CC)(C)C)O)ccc(Cl)cc1F 26303,C(=O)(N1CC(O)CCO1)C1CCCN(C(c2ccnn2C2CC2)=O)CC1 26304,C(C1(C)CCOCC1)=CC(=O)NCC(CNC(CCN(CC(C(C)C)C)C)=O)O 26305,c1(CC)ccc(C(=O)C(=O)NCC(C2CC2)N(C)C(C2(C(F)F)CCCO2)=O)s1 26306,CCC(CC(F)(F)F)C(=O)N1CC2CC3CC2C1C3NC(=O)CCCF 26307,n1(CCC)cc(C(=O)N(CCCNC(=O)CNC(=O)NCC#N)C)cn1 26308,Cc1sc(C(=O)NC2CCC(CCNC(=O)Cc3ccn(C)n3)C2)cc1Br 26309,N1(C(CN(C)C(N)=O)=O)CC(NC(C2(C)CCCC2(F)F)=O)CC12CCC2 26310,c1(O)cc(C)ccc1F.c1(COC)ccc(C(=O)NCC2(CO)CC2)o1 26311,C1(c2n(Cc3cn(CC)nn3)ccn2)CCCCCCC1.c12ccc(s1)CNC2C 26312,N1(C(CSC)=O)CCN(C(C2COCC2C(F)(F)F)=O)C(C(C)C)C1 26313,N1(C(C(C(CC)C)O)=O)CC2(C1)SCCC2NC(c1ccc(CO)cn1)=O 26314,c1(C(CNC(COCC=C)=O)NC(=O)CCCc2ccsc2)ccc(OC)cc1 26315,c1(C(N2CCC3CCN(C(=O)C4=COCCC4)C3C2)=O)cc2cc(F)ccc2[nH]1 26316,c1(C(=O)NC2C3(NC(c4cc(C)nn4C)=O)CCC(C2)C3)cccc2[nH]ncc12 26317,CCCCCC(O)CC(=O)N1CC2CC2C1C(=O)NC(C)C(C)F 26318,Cc1cnc(C(N2CCOC(CNC(=O)C=CC(C)C)C2)=O)nc1 26319,c1(CN=C(NCc2cc(C)on2)NC2CC2C)cn(C)c(=O)nc1O 26320,CCC(CC)(CCNC(=O)C=NOC)NC(C1CCC1n1cccn1)=O 26321,c1(NC(c2cc(I)ccc2-n2cnnn2)=O)ccc2nnn(O)c2c1 26322,c1(C(=O)NC2C(NC(c3c(C)cc(O)cc3)=O)C2)[nH]c2cc(F)cc(F)c2c1C 26323,C(C1=CCN(C(=O)COCC(F)F)CC1)NC(C1C(C)(C(C)C)C1)=O 26324,C(=O)(CCC(C)N(C)C)NC(C(=O)NCC(COC)(C)C)CN(C)C 26325,C1(N(C(C=CCOC)=O)C)CC2(C1)CC(NC(C1(OC)CC(C(F)F)C1)=O)C2 26326,CCCCC(CC)CC(=O)NCC1CC(F)(F)CN1C(=O)C(C)C(C)COC 26327,N1(C(C2(CNC(CC3(C#N)CC3)=O)CC23CCC3)=O)CCC(C2CCC2)C1 26328,C(=O)(CCC(=O)NCC)NCC1(NC(CC=CCC)=O)CCC1 26329,N1(C(C(CN(C)C)NC(=O)COCCCF)=O)CCCN(CCO)CC1 26330,C1(n2cc(C3CCN(C)C3)nn2)C=CCC(C(=O)NCC2CCSC2)C1 26331,C(C(C)(CNC(c1cnc(CC)[nH]1)=O)OC)NC(C(C)OCC=C)=O 26332,CC(C)C(CCNC(c1ccc(N(C)C)cn1)=O)NC(=O)CCN1CCCCC1 26333,c1(C(N2C(CNC(=O)CCC3CCCCC3)C=CC2)=O)ccn2ccnc2n1 26334,N1(C(c2c(C)nc[nH]2)=O)CC(CCNC(=O)Cc2cnc(C(F)(F)F)s2)C(C)C1 26335,N1(C(C(C(C)C)CNC(=O)OC(C)(C)C)=O)CC2CCN(C(=O)CCF)CC12 26336,CCCCC(C)C(=O)NCCCC(O)C(=O)NCCCC(=O)NO 26337,N1(C(C2CC(C#N)(O)C2)=O)CCC2CC(NC(=O)CS(N)(=O)=O)CCC2C1 26338,c1(C(=O)NC2CC(C)(NC(=O)COc3ccccc3Cl)C2)c(O)cccc1Cl 26339,n1(CC(C)C)ccc(C(=O)NCc2cc(C(=O)NCCNC(=O)CO)cs2)n1 26340,CNS(=O)(=O)NCC(=O)NC1COCC1CNC(=O)C(C)NC(N)=O 26341,C(CC(CC)C(=O)NC1CN(C(c2cnn3ccsc23)=O)C(C)(COC)C1)=CC 26342,C1(NC(c2n(CC)ccc2)=O)CN(C(=O)C(C)C2CC2)CCC12CCOCC2 26343,C1(F)(C(=O)NCC(CN(C)C(C2CC23CCOC3)=O)(C)C)CCCCCC1 26344,CC1(C)CCN(C(=O)CN2C(=O)CCCC2=O)CC1C(N1CCC=C(F)C1)=O 26345,C1(NC(N(CC(=O)OC(C)(C)C)CCC)=O)CC2CCC1CC2C(=O)O 26346,c1(C(N(CCN(C(=O)CCc2ccnc(Br)c2)C)C)=O)ccccc1C#N 26347,C1(C)(C(=O)OCC)CN(C(c2cc(C#N)n(C)c2)C(=O)NCC2(C)CC2)CCO1 26348,c1(C(=O)NC2(CC)CCN(C(=O)CCSC)CC2)ccc2c(c1)NCC2 26349,CCC(C)(C)CC(=O)N1CCCC(C(C)(O)CNC(c2cc(CO)oc2C)=O)C1 26350,C1(NC(C23CC(C)(C2)C3)=O)CCC2(CC1)CCN(C(C1CCOC1)=O)C2 26351,Cc1c(C(=O)N(C)CCC2CCCCN2)cccc1Br 26352,c1(OC)c(Cl)ccc(Cl)c1C(=O)NCC(C)NC(c1ccc(C(F)F)o1)=O 26353,C1(C(=O)NCC2CC(NC(=O)CCc3ccccc3)C(O)C2)CCCNS1(=O)=O 26354,Cc1ccc(C)c(C(=O)NC2CC2CNC(=O)C(C)Sc2nncn2C)c1 26355,c1(C2C(C(=O)NC3(c4cn(C(CC)C)nn4)CCOC3)C2)ccc(Br)cc1 26356,N=c1[nH]n(CC(N2CC(NC(=O)CC3CCCCO3)C2)=O)cc1Br 26357,Cc1oc(-n2cccc2)c(C#N)c1C(=O)NCC(O)CNC(C1(O)CCSC1)=O 26358,Cc1ccc(N)cc1C(=O)NCCC1CN(C(c2ccc(=O)n(C)c2)=O)CCO1 26359,C1(SCC)CCCC(N=c2[nH]c(=NCC3(CC4CCC4)CC3)[nH]c3c2CSC3)C1 26360,c1(C(N(c2nc(OC)nc(OC)n2)c2ccc(N)cc2F)=O)ccc2ccsc2c1 26361,N1(C(C(CCC)O)=O)CC2(CCN(C(C3CCCCO3)=O)CC2)CC1C 26362,Cc1cc(C(N2CCC(C)C2CNC(=O)Cn2ccnn2)=O)cc(F)c1 26363,C1(C(=O)NC2(CNC(c3ccc(CC)o3)=O)CCC2)CC(C)CC(C)(C)C1 26364,c1(CC(=O)NCC(C2CC2)NC(C(C)OCCC=C)=O)ccc([N+](=O)[O-])c(N)c1 26365,C=CC(C)CC(=O)N(C1CCN(C(c2cc(C)sn2)=O)C1)CC 26366,N1(C(=O)NC(CC)C(c2nnnn2C)SC(C)(C)C)CC2(C(=O)O)CC2(CO)C1 26367,CCCCC(O)C(=O)N1CC(NC(=O)Cc2cc(C)sc2C)C(SC)C1 26368,N1(C(CC2C(NC(c3n(C)nc(O)c3)=O)CCCC2)=O)CCOC2CCCC12 26369,Cc1ccc(F)cc1C(F)(F)C(=O)NC(C)C(C)NC(C1CC2(CSC2)C1)=O 26370,N1(C(c2n(C)nnc2)=O)CCC(C(=O)NCCNS(N)(=O)=O)C1(C)C 26371,C1(CNC(C=CCCC)=O)CC2CC(C1)N(C(=O)CCc1cccnc1)C2 26372,CC(C)(CCCNC(C1CCC(=O)O1)=O)NC(c1sc(OC(F)F)nc1Cl)=O 26373,c1(C(=O)NC2C3CN(C(CC(C=C)CCC)=O)CC32)c(O)nnc2c1CCC2 26374,N1(C(C2CC(NC(C(C)(C3(C)CC3)OC)=O)C2)=O)CC(C)CC(C)C1 26375,Nc1c(C(=O)NC2CC(NC(C3C4C5CCC(C5)C34)=O)C2)ccc(Cl)c1O 26376,c1(OC)cnc2ncnc(N3CCCCCC3CCO)c2c1 26377,C1(OC)CCC(C(=O)NC(CNC(=O)CCc2cccs2)C2CC2)C1 26378,C1(N(C)C(c2csnn2)=O)CCC(NC(=O)C(O)Cn2cncn2)CC1 26379,C(=O)(CC1COCc2ccccc21)N1CCC(CNC(CSC)=O)C1(C)C 26380,CCCCCCCC(=O)N1CCC(NC(=O)COc2cc(F)cc(F)c2)C12CC2 26381,c1(C(=O)NC2C(NC(c3c(C)onc3C3CC3)=O)CCC2)cccc(S(C)=O)c1 26382,c1(C(=O)NCC(CC)(CC)NC(=O)Cn2cncn2)cc(F)cc(Br)c1 26383,N1(C(C2C(CC)CCC2)=O)CC2(NC(=O)CC3CC4C=CC3CC4)CCC1CC2 26384,N1(C(c2ncc(C)nc2)=O)CCC2(CC1)CN(Cc1nccs1)CCO2 26385,C1(N(C(COCCNC(C(C2CCCC2)OCC)=O)=O)C)COCCO1 26386,c1(CNC(C(c2cc(-c3cnn(C)c3)[nH]n2)N(C)C)=O)nnn(C)n1 26387,CC#CCC(C(=O)NCC(C)(O)CCO)NC(=O)C(C1CC1)SC 26388,C1(OC)(CO)CCN(C(c2c(C)cnn2C)C(=O)NCCSC)C1 26389,C1(NC(CCN(CCC)C)=O)CCCN(C(=O)CCCSC)C1 26390,c1(C(C)C)ccc(C(N2CCC(N(C)C(C3C(C(F)F)C3(C)C)=O)C2)=O)c(O)c1 26391,c1(C(=O)NC(CNC(CC=CC=C)=O)CC=C)cc(=NS(C)(=O)=O)cc[nH]1 26392,c1(C(=O)NC(CC(C)NC(c2ccc(SC)s2)=O)C)ccc2nc(CO)[nH]c2c1 26393,C1(NC(CCC2(CCC#C)N=N2)=O)CCC12CN(C(=O)COC1CC=CC1)C2 26394,c1(CC(=O)NCC2CN(C(c3cc(Cl)no3)=O)CCO2)cc(F)c(F)cc1F 26395,C12(CNC(C(=Cc3ccc(F)cc3)C)=O)CN(C(=O)CC3CCC3)CC1CCO2 26396,C1(NC(c2c(C)noc2)=O)CCN(C(=O)C(CO)c2ccccc2)CCC1CO 26397,S(=O)(=O)(c1ccccc1)NCC(=O)N(C(C)CCNC(C1CCC(C)CC1)=O)C 26398,C(=O)(C1CCCn2ccnc21)NC1CC2(C(NC(CC(C(C)C)(F)F)=O)C2)C1 26399,c1(OC)cc(C(=O)N(C)CC2CCCN2C(c2ccn(C3CC3)n2)=O)sc1Cl 26400,C(=O)(C(CC)CCc1ccccc1)NC1C(CC)CN(C(c2coc(Cl)n2)=O)C1 26401,c1(C(=O)NC2CCCC(CNC(C=CC=CCC)=O)C2)cccc2ncc(C)n12 26402,Cc1onc(C(F)(F)F)c1C(N1CCC(CNC(=O)CN2CCCC2=O)C1)=O 26403,c1(C(N(CCOC)CCNC(C2CC3(CC3)CO2)=O)=O)nc(N(C)C)nc(=N)[nH]1 26404,c1(OC)cc(F)c(C(=O)NCC2CCCCC2NC(C2CC(F)(F)C2)=O)c(F)c1 26405,c1(C(=O)NCC2(O)CN(C(C(C)CC3CC3)=O)C2)cccnc1OC(F)(F)F 26406,CC(C)C(F)(CNC(=O)C(F)C(F)(F)F)C(=O)N1CCC2(CCC2)C1 26407,c1(CC)nc(C(=O)NC2CCC(NC(=O)COCc3cc(C)on3)C2)co1 26408,C#Cc1ccc(CC(N2CCN(C(c3cccnn3)=O)C(CO)C2)=O)cc1 26409,N1(CCCNC(N2C(CC(c3onc(C)n3)(C)C)CCC2)=O)CCCC(C)C1 26410,C1(C(=O)NCCSCCO)C2CC2CN1C(c1[nH]nnc1C1CC1)=O 26411,Cc1csc2ncc(C(=O)NC(C)(CNC(C3(Cl)CC3(C)C)=O)C3CC3)c(=O)n12 26412,c1(NC2CCC(NC(Cc3ccc(SC)cc3)=O)C2)ncnc2[nH]cc(C)c12 26413,N1(C(C(C)=CC)=O)CCCC1CN(C)C(C1(C(=O)OC(C)(C)C)CC1C)=O 26414,C1(C(=O)OC)CC(C)N1C(C1(NC(c2cnc(C(C)C)o2)=O)CC1)=O 26415,c1(C(N2CCCC(N(C(=O)C3=NOCC3)C)C2)=O)ccc2c(c1)C(=O)CCN2 26416,c1(CC)cc(C(N2CC(NC(=O)CC=C(C)C)C(F)C2)=O)cc(O)n1 26417,c1(SC)ccccc1CC(=O)NCC(O)CNC(=O)C(C)O 26418,C1(NC(C(C)(C)SC)=O)CN(C(c2cncc(C(C)(F)F)c2)=O)CC1C(F)F 26419,C1(CC)CCN(C(C2CCC2C(N)=O)=O)C1C(=O)NCCCC1(C)CC1 26420,c1(C(C(=O)NCC(CNC(C2C(CC)CCC2)=O)C)C)ccc2ccccc2c1 26421,C(C(O)CC(=O)N(c1cccc(C)c1)CC)NC(COCCC#C)=O 26422,C1(C(N2C(CNC(C(CC)N(C)C)=O)CCCC2)=O)OC2CCC1CC2 26423,C1(OCCNC(c2coc(O)n2)=O)CCN(C(C2(C(F)(F)F)CCC2)=O)CC1 26424,c1(C(C)C)cn2c(n1)CCC(OC(C1C=CC(NC(=O)OC(C)(C)C)C1)=O)C2 26425,C(=O)(C(C)(C)CC(=O)NCc1nc(CNC(=O)CCc2csnn2)cs1)OCC 26426,C(=O)(C(CCS(C)=O)N(C)C)NC1CCN(C(CCCOC)=O)C1(C)C 26427,C12(CC(=O)NC(C)CNC(C3COC(=O)N3C)=O)CC3CC(C)(C1)CC(C)(C3)C2 26428,C1(NC(C(CC=C)C)=O)CCN(C(c2ccc(CCC)[nH]2)=O)CC1C 26429,c1(OCCC)ccc(C(=O)NC2(CNC(C3SCCCS3)=O)CC2)cc1N 26430,c1(C(N2CCN(C(CNC(C=CCCC)=O)=O)CC2)=O)c[nH]c2cnccc12 26431,c1(C(c2n(C)nnn2)NCc2cnoc2C(C)(C)C)nn(C)cc1I 26432,c1(OC)c(C)cc(NC(C2(O)CCN(C(=O)C(O)C(C)(C)C)C2)=O)cc1C 26433,Cc1ccc(CNC(c2c(C)noc2-c2ccc(Br)cc2)=O)c(OC2CCCC2)c1 26434,C1(C(=O)NCC(C)(O)CNC(=O)C=Cc2ccsc2)CCOCC12CCC2 26435,C(CC(O)C(=O)N1CCC(C)(CC(=O)NCC2CCC(=O)O2)C1)SC 26436,c1(-c2cn(C(C(=O)NCCN(C3CC3)CC)C)nn2)cccc(N)c1C#N 26437,C1(OC)CCCC1CNC(c1cn(CCNC(C2CNC(=O)N2)=O)nn1)=O 26438,c1(OC)c(C(=O)NC2CCC2NC(C23CC(F)(C2)C3)=O)cc([N+](=O)[O-])cc1Cl 26439,C(CCCCCC(=O)N(CC(=O)N(C)C)C)NC(C(C=C)CC)=O 26440,C1(COC)CCCCN(C(=O)C(N2CCSCC2C)=O)C1 26441,CC1CC(NC(=O)C=Cc2ccc(Br)cc2)CN(C(=O)C(C)NC(N)=O)C1 26442,c1(NC(c2ccc(Br)c(Cl)c2)c2n(C(C(=O)OC)C)nnn2)ccc(Br)c(C)c1 26443,C1(C(=O)NC(c2ccncc2)C)CN(C(=O)CN2CCC(F)CC2)C2(CCC2)C1 26444,c1(NC(C)=O)ncc(S(=O)(=O)N2CCCC2c2cc(F)cc(Br)c2)s1 26445,CCC(F)(F)C(=O)NCC1CCN1C(=O)CCN1CCNC(=O)C1 26446,N(C(=NCC1CCCCC1)NCC1CCN(c2ccccc2F)C1)C1C(C)C1 26447,C=CCCCC(C(=O)NCc1cn(C2CC2)cn1)NC(=O)CC1(COC)CC1 26448,CCCC(C(O)C(=O)NC1(C)CC(F)C1)NC(C1(CCC)CC1)=O 26449,c1(C(=O)NCC(C)CNC(=O)CC(C)(C)O)ccc(F)c2ncccc12 26450,C(=O)(CS(=O)(=O)CC(=O)N(C)CC1CCCN1C(=O)C(C)CC(C)C)OC 26451,c1(OC)cccc(CC(O)C(=O)N(C)CC2CN(C(C3CCC(=O)N3)=O)C2)c1 26452,c1(CC)cc(C(N2CCCC2c2ccc(F)cc2)C(=O)NC(C)(C)C)ccc1Br 26453,N1(C(c2cnn(C)c2C(C)(F)F)=O)CCC(NC(C2CC2C(F)F)=O)CC(O)C1 26454,C1(C)(CN(C)C(C2OCCC2C(F)(F)F)=O)CN(c2nnnn2C)CCO1 26455,C1(CNC(C#CC(C)C)=O)C(C2CC2)CCN1C(=O)C=Cc1ccc(Cl)s1 26456,N1(C(CC2CC(OC)C2)=O)CC(NC(C2(CC(C)C)CCCC2)=O)CC1(C)C 26457,N1(C(CC(=O)OC)=O)CCC2C1CCCN2C(c1ccc([N+](=O)[O-])c(C)c1)=O 26458,C1(NC(c2ncc(SCC)nc2)=O)CCSC12CN(C(C1C3CCCCC13)=O)C2 26459,CCCCCC(O)C(=O)NCC1CN(C(=O)C(=O)NCCOCCOC)CCO1 26460,N1(C(c2c(C)cno2)=O)CC2CC(NC(=O)CCOC3CCOC3)C1C2 26461,c1(C(=O)NC2CN(C(=O)C=Cc3cncs3)C2)cc(F)ccc1Cl 26462,C1(C)(C(N(CC(C(=O)OCC)C)C)=O)CCN(C(=O)CC=CCOC)C1 26463,C12(NC(c3ccc(CC)o3)=O)CN(C(c3cc4c(s3)CCC4)=O)C(COC)(C1)C2 26464,C(C#N)(C(=O)C(C)(C)CO)c1ccc(Oc2ccc(C)cc2)cc1 26465,N1(C(C(CC)F)=O)CCc2nc(NC(=O)COCCS)sc2C1.c1nc[nH]n1 26466,c1(C(=O)NCC2(C(=O)OCC)CC(F)(F)C2)cccc(Cl)c1F 26467,CC(C)C(F)(F)CC(=O)NC1CC(CNC(c2ccc(O)nn2)=O)C12CCC2 26468,c1(CNC(C(CC)C)=O)ccc2c(c1)CCN(C(C1(C)CCN(C(C)=O)C1)=O)C2 26469,N1(C(C)=O)CC2COCCC2(NC(c2cccc([N+](=O)[O-])c2Br)=O)C1 26470,C1(C(=O)NC(CNC(C(CC)C2CCC(=O)N2)=O)C)CCC(OC)CC1 26471,c1(-c2occc2)cncc(N2CCN(Cc3csc(-c4cn[nH]c4)n3)CC2)c1 26472,c1(N2CCN(C(=O)OC)CC2)nc(=NC2CCCSCC2)[nH]c2c1COC2 26473,N1(C(C2(C(=O)NC)CCC2)=O)CCC2(NC(c3ccc(N)c(N)n3)=O)CC2C1 26474,c1(CN(Cc2c(C)cncc2)Cc2ncccc2C(=O)O)cc(F)cc(Cl)c1 26475,C1(C(N(C2CN(C(c3cnc(C(F)F)nc3)=O)CC2F)C)=O)CCC(C)(C)CC1 26476,n1(CC(=O)NCCN(C(=O)CSSC(F)(F)F)CCOCCO)cc2ccccc2n1 26477,c1(C(N2CCC(NC(C3(CC)CCNC3=O)=O)C2C)=O)cnc2sccc2c1 26478,C#CC1CC2CCC1N(C(=O)CC1CCC(NC(c3cnn(C)c3CC)=O)C1)C2 26479,CC1(C)OC2(CNC(=O)CN3CCC3C)CC1(NC(=O)C(O)Cn1cncn1)C2 26480,C1(CNC(C2(C)CC(=C)C2)=O)C(C)CCN1c1ccnc(C(C)CC)n1 26481,C1(C)(CNC(C(C)NS(CCC)(=O)=O)=O)COCCN(C(=O)CNC(=O)OC)C1 26482,C1(c2nc(C3(C(C)C4CC4)CC3)on2)(c2nn[nH]n2)CCCCCC1 26483,C1(C(=O)NCC2CC(O)CN2C(c2cn(C)c(C)n2)=O)(COC)CCOCC1 26484,N1(C(c2cnc(OCC)nc2)C(=O)NC2(C)CC2)CC(CO)C2(CC2)C1 26485,C12(CSC)CC(C(N3CCC(C)(CCN(C(=O)CC=C(C)C)CC)C3)=O)(CO1)C2 26486,c1(C(N2C(C)CC(NC(c3cnn(C)c3C3CC3)=O)C2)=O)cc(Cl)ncc1O 26487,C1(CCC)C(C)CCCN1CC1CN(CC(N2CCCC2)=O)C1 26488,C12(CCCC1)C(=O)O2.C1(C(N(C)CC)=O)OCCC1NC(C)=O 26489,CC1CC(C(=O)NCC2(NC(=O)CS(N)(=O)=O)CCCCC2)CCS1(=O)=O 26490,C(=O)(CCCC(F)F)NCC(CCCC)NC(=O)CN1CCCC1C 26491,C1(F)(CNC(c2cnsc2)=O)CC(NC(C2CC2F)=O)C1 26492,C1(C(=O)NCCC(CNC(=O)C(C)O)OC)CCCOCC1 26493,C=C(C)CCCC(=O)NCC=CCNC(=O)C(C)c1cncs1 26494,c1(CCNC(=O)N(C2CCCCC2)CCF)ccncc1Cn1cc(C(=O)O)cn1 26495,CC1CCN(CC(=O)N(CCCN(C)C)CCNC(C2CCSCC2)=O)C1 26496,CCCCCCF.C(CC(=O)CCO)n1cc(CN)nn1.c12nc(cs1)C(=O)N2C 26497,c1(NC(C2C=CC(CC)C2)=O)cc(N(C)CCc2csc(C)n2)ncn1 26498,c1(C(=O)NC2(C)CN(C(c3nc(NC(C)=O)sc3)=O)C2)cncc(N=[N+]=[N-])c1 26499,CCC(C)(CC)C(=O)OCCCC1=NOC(C(N2CCC(C)CC2)=O)C1 26500,N1(CC)CCCCC1C(=O)NCC1CCCCN1C(C1(O)CCCCC1)=O 26501,CC(O)CCCCCC(=O)N1CCN(C(=O)C(F)C(F)(F)F)C2(CCC2)C1 26502,c1(C(C)(C)C(=O)NCC2(O)CC(NC(C3CCCO3)=O)C2)cccc(Cl)c1F 26503,c1(C(=O)NCCC2N(C(C3=CCCC3C)=O)CCSC2)n[nH]c2ccc(F)cc12 26504,N1(Cc2cccc(OC)c2)CCC(O)(C(=O)NC2CCOCC2F)CC1 26505,C1(NC(C(C)NC(CC)=O)=O)CN(C(=O)C(C)(C)N(C)C)CC1(C)C 26506,C1(CNC(Cn2c(C)ccn2)=O)CN(C(=O)CC2C=CCC2)CC1(C)C 26507,c1(C(=O)N(CC(C)C)C(C2CCCC2N2CCOCC2)=O)ccc(N)cc1 26508,c1(C(=O)NC(C2(O)CCN(C(=O)CCc3ccccc3O)C2)C)cnccc1Cl 26509,C(C)(N=c1ccc(Br)c(S(=O)(=O)NCCn2cccn2)[nH]1)c1c(C)cc(Br)cn1 26510,c1(C(C(N2CCCN(c3ccccc3C#N)CC2)C)=O)ccc2c(c1)CCC2 26511,c1(OC(C)C)cccc(F)c1C(=O)NC(C)C(O)Cc1ccccc1 26512,c1(OCC(=O)Nc2nc(C(C)C)nc(C(C)(C)C)c2)c(Cl)cc(Cl)cc1Cl 26513,CCC(CC)(C(=O)NC1CC(N(C)C(C2CC(C)(C)CO2)=O)C1)C(C)C 26514,C1(NC(C(=O)NCCOC)=O)CCC(CNC(=O)CC2CCOC2)C1 26515,c1(OC)cc(CNCC(C(=O)O)OC)cc(I)c1OC 26516,C1(NC(CCC)=O)CCS(=O)(=O)C12CN(C(=O)C(F)(F)C(C)(C)O)C2 26517,c1(OC)cc(C=CC(=O)Nc2ccn(C)c(=O)c2)ccc1OCC(N)=O 26518,c1(CC)cc(C(N2CC(CC(F)C(=O)NCCCc3ncc[nH]3)C2)=O)ccn1 26519,C1(NC(C2CC(C)(CC)C2)=O)CCCC2CN(C(=O)C=Cc3ccccc3)CC12 26520,c1(CCC(=O)NC2(CNC(C3CC(Cl)(Cl)C3)=O)CC2)cnc2ncccn12 26521,c1(NC(C2N(C(C3(C)CC3)=O)C3C(C2)C3)=O)c(F)cc(C#N)cc1F 26522,c1(C(N(CC(C)NC(C2CCCSC2)=O)CC)=O)cc(SC)ccc1Cl 26523,C12(CCCCC1)C(=O)N2.C(=O)(CCOC1CCCC1)N(CC#C)C 26524,CCCCC(CNC(=O)CC1(OC)CCCC1)NC(=O)C(CO)c1ccccc1 26525,Cc1cccc(OCCC(N2CC(O)(C(C)NC(c3c(C)nsc3C)=O)C2)=O)c1 26526,N1(C(CC(=C)C)=O)CCC(NC(c2ccnc(C(F)(F)F)c2F)=O)C(CC)C1 26527,C1(C)(NC(c2c(CNC(CC(C)C3CC3)=O)ccs2)=O)C(C)(C)C1(C)C 26528,c1(N2CCCC(CNC(C3(C=C)CCOCC3)=O)CC2)ncccc1[N+](=O)[O-] 26529,c1(C(C)=O)ncc(C(=O)NCC(C)(C)NC(=O)CC=CCc2ccccc2)s1 26530,C(=O)(C(C(=O)N1CCC(CN(C)C(c2cncn2C(C)C)=O)C1)OC)OC 26531,C1(CC=C)(NC(c2snnc2CCC)=O)CCCN(C(c2ccnc(F)c2)=O)C1 26532,c1(C(=O)Nc2c(C)cc(NC(C3CCC(=O)N3)=O)cc2)c(Br)ccc2c1CCC2 26533,C1(NC(C(c2ccccn2)C)=O)CN(C(c2cccc(Cl)c2)=O)C2CCCCC12 26534,C(CCNC(=O)CCC=CC(C)C)(C(C)C)NC(CCSCC)=O 26535,c1(C(c2n(CCCC)nnn2)NC2CCC3(CC3)C2)sc(Br)c(C)c1C 26536,Cn1nc(C(=O)NCc2csc(CNC(=O)Cc3ccc(=N)[nH]c3)n2)ccc1=O 26537,C(CN=c1cc(C)nc(N2CCOC3(CCSC3)C2)[nH]1)(c1ccc(F)cc1)OC 26538,C1(C(=O)NC23C(CN(C(CC4(C)CCC4)=O)C2)C3)CC2CCCC(C1)C2 26539,c1(C(=O)NCC(CNC(c2ncc(C)c(C)c2)=O)O)ccn2ccccc12 26540,C1(C(=O)NCCOCCNC(Cc2ccc(C(C)=O)cc2)=O)CC2C(C1)C2(C)C 26541,S(=O)(=O)(c1ccc(NC(c2ncc(Br)cc2C)C)c(C#N)c1)NC(CC=C)CC 26542,c1(OC)nccc(C(=O)NC2CCCN(C(=O)C(C)CC(F)F)CC2)c1F 26543,C(=O)(CCCC(=O)OC)N(C1CCN(C(C(C(C)C)OCC)=O)CC1)CCO 26544,c1(CC)nc(N2CC3CC(NC(=O)C(C)C)CC3C2)c(C)c(Cl)n1 26545,C#CC1CCCN(C(C2(C(C)NC(=O)C=Cc3ccoc3)CC2)=O)C1 26546,c1(OC)cc(F)ccc1C(N1CC(C)(C)CC1CNC(=O)CCCC1CC1C)=O 26547,c1(C(N2CCC(NC(CN3C(C)CC3)=O)CC2C)=O)cccc2[nH]ccc12 26548,Cc1ccnc2nc(C(=O)NC3CN(C(C4COC(=O)C4)=O)CC4(CC4)C3)nn12 26549,Cc1ccc(C(=O)NC(C)CCCNC(c2coc(CO)c2)=O)cc1S(N)(=O)=O 26550,C(=O)(CC(C)C(C)(C)C)N1C(CCC)CN(C(=O)CCCc2cnccn2)CC1 26551,N1(C(CC(CC)C)=O)CCC(CNC(=O)C=Cc2ccc(Cl)s2)C12CC2 26552,N1(C(C(COC)OC)=O)CC(C(=O)N(CCCC(C)(F)F)C)CCC1C 26553,C(=O)(C#CC1(C)COC1)NC1CC(F)(CNC(Cc2cc(CC)nn2C)=O)C1 26554,c1(C(N(C2CC(CNC(=O)CSc3nncs3)C2)C)=O)cccc(=O)n1C 26555,c1(C(N2CC(C(C)NC(C(COC)(C)O)=O)OCC2)=O)cncc2[nH]ccc12 26556,CC(C)CC(C)CC(=O)N(C1CCC(CC(C(=O)Nc2nccn2C)=O)CC1)CC 26557,C(=O)(C1=CCCOCC1)NC(CCC)CCCNC(=O)CCN1CCCCC1=O 26558,CCC(C)C(C(=O)N1CCC(n2cc(Cn3cncn3)nn2)C(O)C1)N(C)C 26559,N1(C(Cc2c(C)nn(C(F)F)c2C)=O)CCN(C(C2C=CC=CC=C2)=O)CC(O)C1 26560,C1(N(C)C)CCCN(C(C2C=CCN(C(=O)C=Cc3ccnn3C)C2)=O)C1 26561,C1(C(=O)NCC2CCC(C)CN2C(C2CCCCC2)=O)CC2(COC(=O)N2)C1 26562,N1(C2CN(C(c3c(SC)csc3)=O)C2)CCN(C(=O)OC(C)(C)C)CC1 26563,c1(C(N2C(CC(=O)NC3CC=C(C)CC3)CCC2)=O)ncn2ccccc12 26564,CP(C)(=O)CC(=O)N1CC2(NC(C3CN(C(C4CCCCC4)=O)C3)=O)CC1C2 26565,C1(NC(N(C)Cc2cccnc2)=O)CCCC(C(F)(F)F)C1 26566,c1(NC(c2c(-c3ccc(OCC)c(CO)c3)nccc2)=O)cc(OC)c(C)cc1C 26567,C1(CNC(C(C(C)C)C)=O)CCN(C(=O)CCC2(C)CC2)CC1(F)F 26568,CCC(C(=O)NC(C)(CNC(c1cc(C2CC(F)(F)C2)[nH]n1)=O)CO)C(C)C 26569,N1(C(C(=O)NCCC)CC2CC(F)(F)C2)CCC(C2CCCCC2)CC1 26570,c1(CC(=O)NCCn2cc(CC(CC)(C)O)nn2)cccc(F)c1Cl 26571,C1(NC(=O)COC(=O)CO)CCN(CCNC(c2cocn2)=O)CC1 26572,c1(C(CN2CCC(CCNC(C(COCC)C)=O)C2)O)cccc(S(C)(=O)=O)c1 26573,CC1CC(C)N(C(c2ccns2)=O)CCN1C(c1ccc(CC2CC2)cc1)=O 26574,N1(C(c2cn(C)cn2)C(=O)NCCC2(C)CC2)CCC(CO)C1c1ccccc1 26575,CC1CC(NC(C2CCC2)=O)CCN1C(c1cnn(C2CC2(F)F)c1)=O 26576,c1(C(=O)NCC2(NC(=O)CC(F)(F)F)CCC2)cc2c(nn1)CCC2 26577,n1(CC)cnc2[nH]c(=NC3CC3CC)nc(N3CCCC(OC)C3)c12 26578,C1(CNC(CSc2n(C)ncc2)=O)CC(C)(C)CCC1NC(=O)CSC1CC1 26579,c1(C(=O)NC(CC)CNC(=O)C=CCF)cccc(NC(C)=O)c1 26580,C1(CNC(=O)CCN2CCCCC2)CC(NC(C2(C3CC3)CCC2)=O)C(O)C1 26581,c1(OC)ncc(Cl)c(C(N2CC(N(C)C(c3ccccn3)=O)C(O)C2)=O)c1Cl 26582,c1(C(=O)NC(c2ccc(OCC)c(OC)c2)C)ccc2c(c1)C(CN)CCC2 26583,C1(NC(CSC)=O)CC(NC(=O)C(C)=CC2CC2)C1 26584,C#CC1(CNC(C2(NC(c3ncc(F)cc3F)=O)CCSC2)=O)CCOCC1 26585,c1(OC)ccc(F)cc1CCC(N1CCCC1CNC(c1cc(O)nn1C)=O)=O 26586,C1(C(=O)NCC(C)(C)C#N)CCCC(NC(=O)CC(C)(C)C)CC1 26587,c1(NCC(=O)NC(C(CO)NC(C(F)OC)=O)C)nc(C)nc2sc(C)c(C)c12 26588,c1(CNCCC2CCN(CC)C2)cccc(C(OC)OC)c1 26589,C1(NC(c2cnn(C)n2)=O)C=CCC(C(=O)N(C2COCC2O)C2CC2)C1 26590,C=CCC(CNC(C1(C2CC2)CC1)=O)NC(c1c[nH]nc1-c1ccc(Cl)s1)=O 26591,N1(CC(C)C)CCC(C(=O)NCC(C(C)(C)C)NC(=O)C=CC2CCCO2)CC1 26592,C1(C(=O)NCC2CC2CNC(C2(O)CCOCC2)=O)C2CCCCCC12 26593,CCCC(C#N)C(=O)NCC1(O)CCCN(C(c2c(C)cnn2C)=O)C1 26594,C(=O)(CCC(C)(C)C(=O)N(C)CCN(C(C1CCCCC1F)=O)C(C)C)OC 26595,N1(C(C2CC(=C)C2)=O)CCN(C2CCC(NC(=O)Cc3ncccc3C)C2)CC1 26596,c1(NC(C(C(C)NC(=O)C(F)C(C)(F)F)(C)C)=O)cc2ccccn2n1 26597,N1(C(=O)Nc2cnc(-c3c(C)nc(C)s3)s2)CCc2ccc(Br)cc2C1 26598,c1(C(=O)NC2CN(C(C3C(CC)CCCC3)=O)C2)cc2c(C)ccc(F)c2[nH]1 26599,C(c1ccccc1OC)=CC(=O)NCC1CCC(NC(C(CC=C)C)=O)C1 26600,N1(C(C(CSC)O)=O)CC(C(=O)NCC2(C(C)C)CC2)CC1(C)C 26601,N#Cc1c(Cl)cc(-c2cn(CCNC(C3(O)CCC3)=O)nn2)cc1Cl 26602,CC1(CNC(C2C3COCC23)=O)CCN(C(C2(C(N)=O)CCC2)=O)C1 26603,N1(Cc2cccc(C)c2)CCC(C)C(NC(c2cc(C3CC3)nn2C)=O)C1 26604,C1(NC(C(CC)=CC)=O)CCCC(NCc2cccc(CN3CCCC3)c2)C1 26605,CCC(C)(C#N)C(=O)NCCOCCNC(c1ccccc1-c1nncn1C)=O 26606,c1(OC)ncc(C(N2CC(NS(=O)(=O)C(F)(F)F)CC(F)C2)=O)cc1Br 26607,c1(N(C(N2CC(=C(C)C)C2)=O)C(C)C)cccc([N+](=O)[O-])c1 26608,N=c1nc[nH]n1CC(=O)NCC1CCCC1C(=O)NOC1CC1 26609,N1(C(C(C2CCC2)OC)=O)CC(CNC(=O)CC2(OC)CCCCC2)C(C)C1 26610,N1(C(c2n(CC)ncc2)=O)CCN(C(c2nocc2Cl)=O)C(c2cccnc2)C1 26611,CN1CCCC(C(=O)N(C2CCN(C(=O)CSc3cn[nH]c3)CC2)C)C1 26612,N1(C(c2c(OC)cccc2)=O)CC2CCC1C(CNC(=O)CCOCC(F)F)C2 26613,c1(OCC)cccc(C(=O)NCC(CO)NC(c2cc3scnc3[nH]2)=O)c1N 26614,C1(CC)(NC(C2SCCS2)=O)CCN(C(c2ccc(F)o2)=O)CC1 26615,S(=O)(=O)(CC(=O)NCC1(F)CC(NC(c2cccn2CC)=O)C1)NCC 26616,CCC(CCCC(=O)N1CC2(C1)CC2(F)F)NC(C1(O)CCSC1)=O 26617,c1(CNC(CNC(=O)NC(C)(C)C)=O)csc(C=O)n1.C1(CSC)CC(O)C1 26618,c1(C(=O)NCCN(C2CCCCCC2)C(CC(C)OC)=O)cn(C)nc1Cl 26619,C1(CNC(CC(C=C)C)=O)CCC2(CCC2)CN1C(=O)C(c1ccncc1C)C 26620,C(=O)(C#CC(C)(C)C)NC1(CC(=O)NCc2nnn(CC)n2)CCCCC1 26621,CCS(=O)(=O)Cc1cn(CCCc2nc(-c3ccc(Cl)s3)no2)nn1 26622,C1(c2cn(C(C)C)nn2)C(C)CCN1C(c1ccc(OCS)o1)=O.N(C)C 26623,C(c1ccccc1)=CCCC(N1CCC(N2CCC2)C1)=O.N=c1nc[nH]n1CC(=O)N 26624,c1(OC)ccc(S(=O)(=O)N2CCOCC2C2CC2)cc1CC(=O)O 26625,CCCCCC(F)C(=O)N(CC(N1CCc2nc[nH]c2C1)=O)CCOC 26626,C1(NC(C2CCCC(C(=O)OC)C2)=O)CCCN(C(=O)C(C)n2ccnc2)CC1 26627,c1(NCCCSC(C)(C)C)ccc(C(F)(F)Cl)cc1 26628,N1(C(=O)CC2CCCO2)CC2(C=C(C(=O)N3CC(F)CC(F)C3)CO2)C1 26629,C1(CN(C(=O)CC2CC(F)C2)C2CC2)CCN(C(=O)CC2(O)CCC2)CC1 26630,C1(O)(CC(N2CC(CCCCNC(C3C(C)(C)C3)=O)C2)=O)CCOC1 26631,c1(OCC)ccc(N)c(C(=O)NCC2CCN2C(=O)CCCn2cc(C)cn2)c1 26632,C1(C)(C(=O)NCC2CCC(C(=O)NC(c3ccncc3F)C)C2)CC(C#N)C1 26633,N1(c2nnc(CC)o2)CC(C)CN(C(c2ccc([N+](=O)[O-])s2)=O)CC1C 26634,c1(C(N2CCCC(N(C(c3cc(OC)cs3)=O)CC)C2)=O)cc(C)c(C)cn1 26635,c1(C(N2CCCCC(NC(C(COC)OC)=O)C2)=O)cc2cc(C)[nH]c2cc1Cl 26636,C(=O)(CC1=CCOCC1)NCCNC(C(C)(c1ccccc1)OC)=O 26637,C(=O)(C(C)S(=O)(=O)C(C)C)N1CCC(CC=C)(NC(C2(CSC)CC2)=O)CC1 26638,c1(C(=O)Nc2nc(C(F)(F)F)c3ncnc-3[nH]2)cc(F)cc2nccnc12 26639,C1(CNC(CCC)=O)CCC12CCN(C(=O)COc1ccc(Cl)cc1C)CC2 26640,C(=O)(C(CN(C)C)c1ccccc1)N(CCN(CC)CC)CS(C)(=O)=O 26641,c1(NC(C2CC2C(=O)Nc2cc(Br)cnc2Br)=O)c(Cl)cnnc1Cl 26642,c1(NC(C2(C)CN(C(c3c(C#C)cccc3)=O)C2)=O)cc(Br)c(F)cc1C 26643,N1(C(CCC(C)C)=O)CCN(C(c2cc3n(n2)CCNC3=O)=O)C2COCC12 26644,c1(C(N2CCC(CNC(c3c(CC)scc3)=O)C2)=O)n[nH]c2c1COC2 26645,N1(C(Cc2c(C)non2)=O)CCC2(C1)CN(C(C1CCCS1(=O)=O)=O)C2 26646,N1(C(C(CC)C)=O)CCC2CN(C(=O)C3=C(C)OCC3)CC2CC1 26647,N1(C(C(CC(C)C)N(C(=O)C2=CCCCC2C)C)=O)CC(O)C2(CCCC2)C1 26648,C(=O)(C(F)(F)C(C)(C)O)N1CC(CC(C)NC(=O)C(=Cc2c[nH]cn2)F)C1 26649,C1(F)(CNC(C(=O)N(C)C)=O)COCCN(C(C2COCC2(C)C)=O)C1 26650,C#CCC(C)(CC)C(=O)NCCN(C(c1cnc(C2CCC2)o1)=O)C(C)C 26651,C#CCC(C(=O)Nc1ccc(C2CC2)cc1)NC(C)C(=O)OC 26652,Cc1c(O)ccc(C(N2CC(F)CC2CNC(C2(C)CCN(C)C2=O)=O)=O)c1C 26653,c1(C(=O)NCC23N(C(C4C(C)(C)CCC4)=O)C(CC2)CC3)ccsc1S(C)(=O)=O 26654,c1(C(=O)NC(C(C)NC(=O)C(F)OC(F)(F)F)CO)ccn(C)c1C1CCC1 26655,c1(NC(C2CN(Cc3cccc(F)n3)CCC2O)=O)cccc2nc(O)ccc12 26656,CC1(C)CCN(C(c2cncnc2)=O)CC1NC(c1cc(-c2ccoc2)[nH]n1)=O 26657,c1(C(N2CCC(N(C(=O)CCCCC#N)C)CC2)=O)cc2ccncc2cc1F 26658,c1(-c2nc(Cc3ccccc3)oc2)nc(Cn2ccnc2)nn1-c1ccccc1 26659,c1(C(=O)NC2C(CNC(C(n3ncc(C)c3)C)=O)C2)cncnc1C(C)C 26660,C1(CNC(=O)Cc2ccsn2)CCCC(NC(c2ccsc2C(F)F)=O)C1 26661,N1(C(c2c(C)con2)C(=O)NC(c2ccccc2)C)CC(C)(C)C1C(C)C 26662,C1(C(=O)NC(c2ccsc2)C)CN(C(=O)C(=O)NC2CC2)CCC1(C)C 26663,c1(OC)cc(NC(C2(CNC(=O)COC(C)C)COC2)=O)cc(Br)c1 26664,C12(C(=O)NC3C(NC(CC=CC=C)=O)CCCC3)CCC(CC)(C1)OC2 26665,C(C(=O)Nn1cnnc1)(C(C)CC)NC(c1cc(=NC)[nH]cc1)=O 26666,C(=O)(CCC(C(C)C)NC(c1ocnc1C(C)C)=O)NCC(C1CC1)OC 26667,C1(N(C(COCCCCC)=O)CC)CCN(C(C2CCOC2CC)=O)C1 26668,N1(C(C(C=C)O)=O)C2CCC1C(F)C(NC(=O)Cc1cccc(C)c1)C2 26669,N1(C(c2c(C)n(C)nc2)=O)CCC2(CCCN2C(=O)CCCc2cccs2)C1 26670,CC(C)CC(C(=O)NC(CNC(C1(n2ccnn2)CC1)=O)C(C)C)N(C)C 26671,C1(C)(CC)CC(C(=O)NC2CC(C(C)NC(c3sc(C)nc3OC)=O)C2)CCO1 26672,c1(C(=O)NC(CC)CNC(=O)C(C(C)C)NS(C)(=O)=O)ccc2nc(C)oc2c1 26673,S(=O)(=O)(c1ccc(Br)cc1N(C)Cc1cccc(Cl)c1)NCC1OCC(C)C1 26674,N1(C(CCC(=O)NCC)=O)CC(NC(C2CC=CC2)=O)CC(F)C1 26675,c1(C(=O)NC(C)CCNC(C2(CO)CC2)=O)cn(C)cc1C(F)(F)F 26676,C12(C(=O)NCC3N(C(c4c(C)n[nH]c4C)=O)CCC3)CCC(CC1)C(C)O2 26677,N1(C(Cn2ccc(C)n2)=O)CC(C(N2CC(n3ccnc3)C2)=O)C2(CC2)C1 26678,c1(C(=O)NCC(CC)NC(=O)C(O)CC2CC2)cc(F)n(C)n1 26679,N1(C(CCC=C)=O)CC2CC(C(=O)NCc3cccnc3OC)C(C2)C1 26680,C(C1=CCN(C(=O)C2=CCCOC2)CC1)NC(c1ccc(C(N)=O)[nH]1)=O 26681,N1(C(C2(F)CN(C(C(C(C)C)SC)=O)C2)=O)CC2CN(C)CC2C1 26682,c1(C(N(CC(O)CNC(=O)CN2CCNC(=O)C2)C)=O)cc2nc[nH]c2cc1F 26683,N1(C(c2ccc(N)c(F)n2)C)C2CCC1CC(N1CCN(CC(F)(F)F)CC1)C2 26684,C(=O)(C(C)(CC)C(=O)OCC)NCCC1CCN(C(CC=CC=C)=O)C1 26685,c1(C(=O)OCC)cnn(CCNCCC2OCCC2C)c1 26686,CCC(CC(C)C)C(=O)N1CC(C(=O)NCc2ccccn2)C2(CC2)C1 26687,Cc1ccc(Br)c(C(=O)NC23CC2CN(C(=O)COCC(C)(C)C)C3)c1 26688,C1(CNC(c2c(C)nco2)=O)CN(C(C2CC2c2sccc2C)=O)CC12CCC2 26689,c1(NC(C(=O)NCCCCSC)=O)ccc(Br)cc1SC 26690,C1(C2(O)CN(C(c3nccc(Cl)c3F)=O)C2)(CNC(C2CCC3(CC3)C2)=O)CC1 26691,CN1CCCC(C)(C(N2CC(NC(C3CCCN3N=O)=O)C(C)(C)C2)=O)C1 26692,C1(OC)CC(C(=O)OC)N(C(=O)NC(C)C(C)SC)C1.C(C)(C)O 26693,c1(CC)[nH]c(C(=O)NCC(C)(CO)NC(c2cc(C)nn2C)=O)nc1Cl 26694,c1(COCC)cccc(-c2cn(C3CCC(C(=O)NOC)CC3)nn2)c1 26695,C1(CNC(C(=O)NC2C(c3n(C)nnc3)C2)=O)CCC(C)(C)CO1 26696,c1(C(=O)NCC2(CSC)CCC2)cccnc1-c1nc(C2CCC2)no1 26697,c1(CC)noc2ncc(C(=O)NC3CC4CC(C3)N(CC(C)OC)C4)cc12 26698,Cc1cnc2n1CC(C(N1CC(N(C)C(C3SCCCS3)=O)C3(CC3)C1)=O)CC2 26699,N1(C(=O)CC2(O)CCOC2)Cc2n[nH]cc2C1C(=O)N1CC2CCCC2C1 26700,c1(C(N2C(C(C)NC(C3CC3C(C)(F)F)=O)CCC2)=O)c[nH]c(=S)cn1 26701,c1(OC)ccc(C=NOCC(=O)NC2CC2CNC(=O)Cc2cc(C)cs2)cc1 26702,c1(OC)cc(C)c(C(N2CC3CC3(CNC(C3(C)CC4CC4C3)=O)C2)=O)cn1 26703,N1(CC(=O)NC(C(=O)NCCC(=O)NC(C)C)C2CC2)CCCCC1=O 26704,c1(C(N(C(C(=O)NCC=C)C2CCN2C(=O)OC(C)(C)C)C)C)ccc(F)cc1 26705,C1(NC(c2cncc(C)c2Cl)=O)CCN(C(=O)CCOCC2CC2)CC1(C)C 26706,Cc1nn(C)cc1C(=O)N(CCCNC(=O)C(C)Sc1ccc(Cl)cc1)CCO 26707,CC(C(O)C(=O)NC1(CCNC(c2cccnc2S)=O)CC1)c1ccccc1F 26708,c1(NC(CC2CCCN(C(C(CCCC)O)=O)C2)=O)c(I)cc([N+](=O)[O-])cc1I 26709,N1(C(C(C2CCN(C(c3cnn(C)c(=O)c3)=O)CC2)C)=O)CC2(CNC(=O)C2)C1 26710,C1(C(N(C)CC2N(C(CCc3cc(OC)no3)=O)CCC2)=O)CC(C)OC(C)C1 26711,N1(C(c2c(F)ccc(C)c2O)=O)C2CCC1CC(F)(CNC(C1CC13CC3)=O)C2 26712,C1(C(=O)NC(CN(C(c2c(C)scn2)=O)C)(C)C)CCCC(F)C1 26713,N1(C(CNC(COC)=O)=O)CCC(c2n[nH]c(CNC(=O)C=CC3CC3)n2)CC1 26714,C(=O)(C(O)CC(C)(C)C)NC1(C)CCN(c2snc(C(C)(C)OC)n2)C1 26715,C1(NC(CSC)=O)CCN(C(=O)CCNC(C)=O)CC1C(N)=O.C1C(=O)N1 26716,N1(C(C(C(C)C)NC(Cc2cc(C)nn2C)=O)=O)CC2(C1)CN(C)CCO2 26717,c1(C(=O)NC23CCCC(NC(CC=C)=O)(C2)C3)ccc(Cl)c(F)c1N 26718,c1(N2CCCC(CN(C(C3(OC)CCCOC3)=O)C)C2)cccc(F)c1[N+](=O)[O-] 26719,C1(C(=O)NCC2(CCOC)CCCC2)(CNC(=O)COCCCF)CC12CCC2 26720,c1(C(=O)OC)cc(C(=O)NCC2(CN(C)C(c3ccn(C)n3)=O)CC2)nn1C 26721,N1(C(c2ccc(C)n2C)=O)C2CCC(C2)C1CNC(=O)C(C)OCCC(C)C 26722,c1(C(=O)NCCN(C(=O)Cc2cc(Cl)ccc2F)C)cncc([N+](=O)[O-])c1 26723,N1(C(C)C(=O)NCCC2CCCN2C(=O)COC(C)(C)C)C(=O)CCC1=O 26724,C(=O)(C1OCCc2ccccc21)N(CCNC(CC(C)OC)=O)C(C)C 26725,C=Cc1ccc(C(=O)NCC(F)CNC(=O)C(C)(C)C#N)cc1 26726,C1(C(=O)NCC2C(C)OCC2)CN(C(C2CC(N=[N+]=[N-])C2)=O)CC12CCC2 26727,Cc1cc(C(N2CC(NC(=O)C(=O)NCC(F)F)C2)=O)c(C)cn1 26728,C1(CN(C(C(C)NS(CC)(=O)=O)=O)C)CN(C(c2cc(Br)n[nH]2)=O)CCO1 26729,C#CCC(CC(=O)N1CCCC1C(C)CC)NC(c1cc(O)ccc1F)=O 26730,N1(C(CCCC(C)C)=O)CC2(CCN(C(c3cc(C(F)(F)F)n(C)n3)=O)C2)C1 26731,c1(CC(C(=O)OC2CCN(CC(=O)OC)C2)O)ccc(F)cc1Cl 26732,C12(NC(c3c(C)nsc3)=O)CCN(C(c3cnc(N)cn3)=O)CCC1C2 26733,C1(CNC(COCc2onc(C)n2)=O)CCCCN1C(C1COCC1C(F)F)=O 26734,CCCS(=O)(=O)C(C)C(=O)NC(C)CCNC(=O)Cn1nnc(=N)[nH]1 26735,CC1CC2(CC2)CN1C(C1OCCC1CNC(=O)Cc1cccnc1O)=O 26736,S(=O)(=O)(c1ccc(I)cc1)N(C1CCCN(C)C1)C.c1(N)ccc(NC=O)cc1 26737,N1(C(C(CCC)OC)=O)CCC2(CC1)CC(NC(=O)CC(C)CC)C2 26738,C1(NC(C2(CC#C)CCCO2)=O)CCC(O)CN(C(c2cc(C)no2)=O)C1 26739,C=CCCCC(C(=O)NCC1CN(C(=O)OC)C1)NC(=O)C(C)CC(=C)C 26740,CC(C)(C)CC(O)C(=O)NC(c1cccc(O)c1)CO 26741,c1(C(C)NC(=O)NNC(=O)c2nccn2C)nc2ccccc2o1 26742,N1(C(c2c(CC)ccs2)=O)CCOCC1CNC(=O)C(C)Oc1ccc(F)cc1 26743,c1(C(N2CC3N(C(CCCCSC)=O)C(CC3)C2)=O)n[nH]c2c1CC(F)(F)CC2 26744,C(CN=c1cc[nH]cc1S(=O)(=O)N1CCC(C)(CO)C1)N(C)N(C)C 26745,C(CC(=O)NC1CC(NC(=O)C(C)=C2CCC2)C1)=CCC 26746,c1(C(=O)NCC(C)CNC(C2COCC3(CCC3)O2)=O)cccc2nc(O)[nH]c12 26747,c1(C(=O)NC2(C)CCN(C(C(C(C)(C)O)F)=O)C2)cc(O)c2ccoc2c1 26748,c1(C(CCO)Cc2n(C(C(=O)OC)C)nnn2)ccc(OC(F)F)cc1.C(CCO)N 26749,C1(C(=O)NCCC=CCCC)CN(C(=O)CCc2cnoc2)CC1CCOC 26750,N1(C(c2c(COC)cco2)=O)CC2CC3CC2C1C3NC(c1cc(CO)[nH]n1)=O 26751,C1(NC(C2C(C)=CCS2)=O)CCN(C(=O)CCc2ncnn2C)CC1O 26752,c1(CCOC(C)=O)nc(-c2cccc(Cl)n2)nn1CC(C)C 26753,C(=O)(CC(F)(F)C(F)F)N1C(C(=O)NCC(CCOC)(C)O)CCCC1 26754,C1(C(N(C2(C(=O)NC3(CCO)CCOC3)CC2)C)=O)CCCCC1(F)F 26755,C(CCCCC(=O)NCC(CC)NC(=O)CC1CN(C)C1)OCC 26756,C1(NC(=O)CCC2CCCCO2)CCN(c2nnc(C(F)F)o2)CC1O 26757,Cc1cccc(C(N2CC(CNC(=O)Cc3ccc(F)cc3)C3CC23)=O)n1 26758,C=Cc1cc(C(=O)NCC(CNC(c2cc(C#N)on2)=O)C(F)(F)F)cc(F)c1 26759,Cc1cn2cc(C(=O)NCC3(CNC(c4cn(C)nc4C)=O)CC3)sc2n1 26760,c1(CCNC(=O)NC(c2ccccc2Cl)C)c[nH]c2ccc(O)cc12 26761,Cn1cnc2c(C(=O)Nc3cccc(Cc4ccc(C#N)cc4)c3)ccnc12 26762,CCC(CCOC)C(=O)N1CC(OC)C(C(=O)NCCCCN(C)C(C)C)C1 26763,C1(COC)(CNC(=O)Cc2ccccc2C)CCCN1C(=O)C(C(C)C)NC=O 26764,N1(CC(=O)NCCOCC)CCN(C(c2cnc(N(C)C)cn2)=O)C(C)C1 26765,CC1(C)CN(C(C2CCCCS2(=O)=O)=O)CCC1NC(c1cc(F)cnc1Cl)=O 26766,c1(C(=O)NCCC(=C)CNC(=O)CCCN=[N+]=[N-])ccc(S(=O)(=O)C(C)C)cc1 26767,N1(C(=O)C2=CCCOC2)CCC(C2CCN(C(c3cc(O)nc(O)n3)=O)CC2)C1 26768,Cn1cc(CNC(=O)C(C2CC2)NC(c2cnns2)=O)nn1 26769,C(=O)(C1=CCC(C)CC1)NC(C1N(C(C(CC(=C)C)C)=O)CCC1)(C)C 26770,c1(COC)ccc(C(=O)N(CC(O)CNC(c2cc(C)ccc2O)=O)C)cc1F 26771,C1(NC(C(CC=C)C)=O)CN(C(c2cccc(F)c2NC)=O)Cc2ccnn2C1 26772,N1(C(c2c(CC)c[nH]n2)=O)CCCCC1C1(NC(c2ccc(C)n2C)=O)CC1 26773,N1(C(CS(N)(=O)=O)=O)CCC2(CCCC2CN=c2cccc(C(F)(F)F)[nH]2)CC1 26774,C1(NC(CC(CN(C)C)O)=O)CCN(C(c2cc(F)ccc2Cl)=O)C12CC2 26775,C(=O)(C1=CCCCC1)NC(CNC(c1c(OC)csc1)=O)C(C)C 26776,C=CCC(C)C(=O)N1CCOC(CCCNC(=O)CCc2nncs2)C1 26777,c1(C(C(=O)N(CCCNC(CC(C)CN(C)C)=O)C)O)ccc(Cl)c(Br)c1 26778,c1(C(=O)NCC(CNC(c2ccn(CC(C)C)n2)=O)F)cccc2c1CCOC2 26779,c1(C(N2CC(C(C)NC(=O)CC(O)C3CC3)OCC2)=O)cc(Cl)ccc1N 26780,C(C(=O)NNC(=O)C1CCCCC1)C1(OCC)CCOC1 26781,C1(C(=O)NCC=CC(=O)N(CCCCC=C)C)CC2(CC2)CO1 26782,N1(CC)C(=O)CCC1CC(=O)NC1CN(C(C2(CC)CC2)=O)CC1OC 26783,C(=O)(CCCC(=O)NC(C)C)NCC12CC(NC(C3N(C(C)C)CCC3)=O)(C1)C2 26784,N1(C(C2C(=C)CC2)=O)CCN(C(c2ccc(C(C)(C)C)cc2)=O)CC1CO 26785,c1(C(N(C2CCN(C(=O)COc3cccnc3)C2)CC)=O)ccc2cccnn12 26786,c1(C(N2CC(NC(C3C(C)(C)CC3)=O)CC3(C2)CC3)=O)[nH]c2ccccc2c1Cl 26787,CC(C(=O)NO)NC(c1nc(CO)cs1)c1nnnn1C1CC1 26788,c1(CC(C(N2CCC(CNC(C3CC(CF)C3)=O)C2)=O)O)cc(Cl)cc(Cl)c1 26789,C(=O)(CS(=O)c1ccc(Cl)cc1)NCC12CCCC(NC(=O)OC(C)(C)C)(C1)C2 26790,c1(CC(N2C(C(C)NC(C(CC#C)(C)C)=O)CCCC2)=O)c[nH]c2ncccc12 26791,C1(C(=O)NC(CCC)C)CCCCCC1NC(c1ncoc1C)=O 26792,Cc1snnc1C(=O)N(CCNC(C1CC(C(F)(F)F)CO1)=O)C1CC1 26793,N1(Cc2cc(C)sc2C)CC2(CCC(CNC(C3(C(F)F)CCOCC3)=O)O2)C1 26794,c1(C(=O)NC(C(=O)N(C(C=C)C2CC2)C)CC2CCC2)cc(C)oc1C 26795,c1(CNC(CC)=O)ccc(CN(C(=O)CC=CC(C)(C)C)C)cc1 26796,c1(C(=O)NC2CN(C(Cn3nnc(C)n3)=O)C(C)CC2)cnn2ccc(O)nc12 26797,N1(C(C(COC)N(C)C)=O)CC(CNC(=O)Cc2c(C)n[nH]c2C)C(C)C1 26798,c1(C(=O)NCCNC(C(N2CCCC(O)C2)C)=O)c(Cl)cc(Br)cc1Cl 26799,c1(CC(=O)NCCCN(C(=O)CNS(C)(=O)=O)C(C)C)nccc2ccccc12 26800,C1(NC(=O)CC2CCCN2C(=O)CCc2nc(O)n[nH]2)CCOC12CCCC2 26801,c1(CC(CNC(CCOC(C)=O)=O)NC(=O)COc2ccsn2)ccccc1 26802,C(CC(C)(C)C#N)(c1n(CCC2(C)CC2)nnn1)NCCC(=O)NCC(F)(F)F 26803,COn1cnc(C)c1C(=O)NC1CC(=O)N(C2CN(C(C3CC3C#N)=O)C2)C1 26804,n1(CC)ncc(Cl)c1C(=O)NCC(O)CN(C)C(C1CC1C(C)(C)C)=O 26805,N1(C(CSCCC(C)C)=O)CCCCCCC1C(=O)N(C)CC1CC1C 26806,c1(OC)cc(Br)c(NC(C2CC2NCc2ccc(O)c(O)c2O)=O)cc1C 26807,C(=O)(C(C(C)(C)C)N1CCNC1=O)N1C(C)C(NC(c2cc(N)ccn2)=O)CC1 26808,n1(-c2ccc(C)c(F)c2)nnc2c1CN(C(=O)CC1=NNC(=O)C1)CC2 26809,c1(C(N2CCC(C)(N3CCCC3)C2)C(=O)NCC=C)cc(Cl)cc(Cl)c1Br 26810,O=S(=O)(c1ccc(NCCCC2CCC2)cc1Br)NC1CC2OCCCC12 26811,Cn1nnc2c1CCC(C(=O)NCC1(C)CC(NC(=O)CCOCC(F)F)C1)C2 26812,CC1CN(C(=O)CCc2cccc(C#N)c2)C(C)CN1C(=O)CCc1nc[nH]n1 26813,c1(CC(N2C(CNC(C(C)CC(C)(F)F)=O)CC2)=O)cc(F)cc2c1OCOC2 26814,C(=O)(CC(C)CF)NC(C)CCN(C)C(c1c[nH]nc1-c1cnn(C)c1)=O 26815,N1(C(c2c(CNC(C(C)OCOC)=O)c[nH]n2)=O)CC2(C1)OC(=O)NC2C 26816,C=CCC(C)(C)CNC(c1cnccc1OC)c1nnnn1CCC(=O)OCC 26817,CN=c1[nH]c(=NCC2(C)COc3ccccc3O2)[nH]c(=NCC2CCOCC2)[nH]1 26818,CC(CC(=O)N1CCN(C(=O)C(C)(C)N=[N+]=[N-])CC12CC2)CC(C)(C)C 26819,C1(C(=O)NCC(=O)OCC=C)CC12CC(NC(c1ccoc1)=O)C2 26820,N1(C(c2c(C)sc(O)n2)=O)CC2COCC2(C(=O)NCC(C)CO)C1 26821,Cc1cc(C(=O)N(CCC(=O)N2CCC2C(N)=O)CCCO)nc(O)c1 26822,Cc1nc(O)nc(C)c1C(=O)NC1CCCC1CNC(c1ccc(N)c(Cl)n1)=O 26823,CC1CN(C(=O)Cc2csc(Cl)c2)CCC1CNC(=O)CCCCN1CCCC1 26824,C(=O)(CCCC(=O)NCc1cnc(Cl)cc1F)NC 26825,CC1CN(C(=O)Cc2c(F)cccc2Cl)CCC1NC(c1cc(C(F)F)no1)=O 26826,C1(F)(C(=O)NC(C(C)C)CNC(c2csc(CO)n2)=O)C2CCCC12 26827,N1(CCN2CC(CC)C(C)C2)CCCC(NC(=O)OC(C)(C)C)C1 26828,c1(CN2CC(C(N)=O)C2)cc(C(F)(F)F)cc(N=c2[nH]c(Cl)ncc2F)c1 26829,N1(C(C2CC(F)(F)C2)=O)CCCC(NC(C2(CC3CC3)CC2)=O)C1 26830,C=C(Cl)CCC(=O)NC1CCN(C(c2cncc(OC)n2)=O)C1 26831,N1(C(C(C)C=Cc2ccccc2)=O)CC2CCC1C(NC(=O)C(C)(F)F)C2 26832,N1(C(C2C(CC)C2)=O)CCC2(CC1)CC(NC(c1cc(Br)nn1C)=O)C2 26833,c1(C(N(CCCNC(=O)C(O)C(F)(F)F)C(C)C)=O)ccnc2c1CCO2 26834,C(=O)(C(CC(C)C)C(C)C)NC(C1CCN(c2nc(COC)nc(C)c2)CC1)C 26835,c1(C(=O)NCC2(O)CN(C(=O)CCc3cn[nH]c3)C2)csc2cccc(F)c12 26836,c1(C(N2CC(C(C)=O)(CNC(C3CCCC3(F)F)=O)C2)=O)cccc(=O)n1C 26837,c1(C(N2C(C)(CNC(C(CCCC)C)=O)CCC2)=O)cn2nc(OC)ccc2n1 26838,CC1CC(C(=O)NC(C2CCN(C(c3cc(C(F)(F)F)no3)=O)CC2)C)=NO1 26839,N1(C(c2c(C)nc(C(F)(F)F)o2)=O)CCC2C(C1)CN2C(=O)Cn1nnc(=O)[nH]1 26840,C1(CC)CC(C(=O)N(CC(C)(C)NC(c2ccc(C3CC3)cc2)=O)C)CC(=O)N1 26841,C(=O)(C(C)(F)F)NCC(CNC(C(C1CCCC1)NC(=O)OC(C)(C)C)=O)O 26842,c1(C(N2CCCC(NC(C(CC)NC(C)=O)=O)C2)=O)cc2cccnc2[nH]1 26843,CCC1=NOC(CC(=O)NCC2C=CCN2C(c2csc(C)c2)=O)C1 26844,Cc1ncc(C(=O)NC(C2CCCC2)CNC(=O)C(F)Cc2ccccc2)[nH]1 26845,N1(C(c2c(CC#N)ccs2)=O)Cc2nccn2CC(NC(C2CN(C(N)=O)C2)=O)C1 26846,c1(C(C(=O)NCC(CNC(COC(CC)(C)C)=O)C)C)cccc(F)c1 26847,c1(CC(=O)NCCCC(C)NC(C2OCCCO2)=O)c(Cl)cccc1Br 26848,O=C(CN=c1cc[nH]cc1)NCCC(O)CNC(c1ccc(O)nn1)=O 26849,N1(C(COCC)=O)CCN(C(C23CCC(CO2)C3)=O)CC1C1CC1 26850,S(=O)(=O)(c1ccc(I)cc1)N1CC2CN(S(=O)(=O)CCCCCl)CC21 26851,c1(NC(CC2CCN(C(c3cccc(C)c3)=O)C2)=O)cc(Br)c(Cl)cc1F 26852,C1(CC(=O)NC2(CC=CC(=O)NCCCOCC=C)CCC2)CCOC1(C)C 26853,C(=O)(C(C#N)C(=O)c1c[nH]nc1C(F)(F)F)Nc1c(OC)cccc1 26854,c1(CC(N2CC3CCN(C(COCCC#C)=O)C3C2)=O)oc2ccccc2c1C 26855,CCC(C)(CC1CCCCC1)C(=O)N1CCN(C(=O)C(F)F)CC1 26856,c1(C(=O)NCC2C(NC(c3ccc(-c4ccccc4)[nH]3)=O)C2)ccccc1F 26857,N1(C(C(C#C)(C)C)=O)CCC2CCN(C(C3CNC(=O)C3)=O)C2C1 26858,C=CC(C)(O)CCCC(C)C(=O)N1CCCN(C(c2cc(Br)no2)=O)CC1 26859,C(=O)(C1=C(C#N)CCC1)N1CC(C(=O)NC2CCN(C(C)=O)C2)(CC)C1 26860,c1(C(CC(=O)Nc2cncc(Cl)c2)NC2C(OCC)CCC2)ccc(F)c(F)c1 26861,c1(C(N(C)CCNC(=O)CSCC(F)(F)F)=O)cccc2c1COC2 26862,C1(C(N(CCN(C(Cn2cc(C(=O)OC)nc2)=O)C)C)=O)CCSC(C)C1 26863,C(c1cccnc1)=CC(N1C(C(C)NC(C2CC=CCC2)=O)CCC1)=O 26864,C(CCC(C)(F)F)N(C(=O)CN(C(=O)CC1CC2CC2C1)C1CCC1)C 26865,C12(CNC(=O)C=Cc3ccco3)CC1CN(C(c1nccnc1C(F)(F)F)=O)C2 26866,C(CN=c1[nH]c2c(c(=NCCCC3CC3(Cl)Cl)[nH]1)CC(C)CC2)c1nc(C)sc1 26867,O=C(Nn1ccnn1)C1C(c2ccccc2O)C1(F)F 26868,C(=O)(C(CC(C)C)CC(C)C)N1C2(CNC(C(CC=C)(C)C)=O)CC(CC)(C1)C2 26869,C=CCC(Cc1ccccc1)C(=O)NC(CNC(=O)CCC=C(C)C)CO 26870,C(CC1=CCN(C)CC1)NC(C1(CC#C)CCN(C(C2CCN(C)C2C)=O)C1)=O 26871,Cc1ccc(C(=O)CCC(=O)N(C)CC2CN(C(c3cnccn3)=O)C2)cc1 26872,Cc1onc(C(=O)NC2CCN(C(c3cnn(CC(F)F)c3C)=O)C2)c1[N+](=O)[O-] 26873,Cc1cc(C(=O)NCC2CN(C(c3ccc(F)cc3)=O)CCC2C)cc(C)c1O 26874,C#CCCCC(=O)N1CCN(C2CN(Cc3cnc(Cl)nc3)C2)CC1 26875,C(=O)(C(C)C(O)C(C)CC)N1C2C(C(=O)NCCCCC)CC(C=C2)C1 26876,C1(CNC(=O)CSc2cn[nH]c2)COCCN(C(=O)CNc2ccccn2)C1 26877,N1(C(c2ccc(NCC=C)cc2)=O)CC(CC)OCC1C 26878,N1(C(c2c(C)ccnc2)=O)CCC(NC(=O)C(F)(F)c2csc(Cl)c2)C(O)C1 26879,c1(NC(C(c2cc(C)ccc2I)N(CCSC)C)=O)c(C)cccc1C 26880,C1(C)(C(=O)NC2CCC(N(C(C=C(C)Cl)=O)C)C2)COC(=O)OC1 26881,CCC(C)C(C)C(=O)N1CCC(CNC(=O)CC(C)NC(=O)C(C#N)CC)C1 26882,C(C1=NOC2CN(C(c3cc(O)nc(O)n3)=O)CC12)NC(=O)C1=CCS(=O)(=O)C1 26883,N1(C(C(C2CC2)OC)=O)CC(CNC(=O)CN(CC(=O)NC(C)C)C)C2(CC2)C1 26884,C(CC(=O)NC1CCC1C(=O)NC(C)C(C)n1cccn1)(OCC)OCC 26885,CCC(C)C(C(=O)NCCNC(=O)C(c1ccc(C(F)(F)F)cc1)(C)C)N(C)C 26886,N1(C(CCCCOCCC=C)=O)CC2(C1)C(NC(=O)C(O)C1CC1)CCS2(=O)=O 26887,Cc1cccc(C(C)C)c1C(N1CCC(CNC(=O)CC2COC(=O)N2)C1)=O 26888,CCC(C(=O)NC(CNC(=O)C(C)C(=O)N1CCOCC1)(CC)CC)C(C)C 26889,CCC(C)(C#N)C(=O)NCCC(=O)NCC1CCCCN1C(c1csnn1)=O 26890,C1(C(=O)NCC(c2ccccc2)NC(=O)Cc2ccoc2)CCCCO1 26891,N1(C(=O)CC2C=CCC2)CCN(C(=O)Cc2ccoc2)C(c2ccccc2Cl)C1 26892,Cc1cc2cc(C(=O)NC34COC(C3)C(NC(=O)C(O)C(C)C)C4)c(Cl)cc2[nH]1 26893,C1(C(=O)NCC2N(C(CC3(C=C)CC3)=O)CC(C)CC2)(CO)CC2CCC1CC2 26894,N1(CC)CC(C(=O)NCC(C2CC2)N(C(=O)CN2C(=O)CNC2=O)C)CC1=O 26895,O(P(C)(=O)CNC(C1(OC)CCN(C(=O)C(C2CC2)OC)C1)=O)CC 26896,C1(C(=O)NCCCN(C(c2coc(CO)c2)=O)CC)CC(C(F)(F)F)CO1 26897,C1(NC(C2CCC3CC23)=O)CN(C(c2cccc3[nH]ccc23)=O)CCC12CCC2 26898,N1(C(Cc2cc(OCC)no2)=O)CCCCC(CNc2cc(OC)cc(C)n2)C1 26899,C(C(CC(C)C)NC(=O)C(C)Oc1ccccc1OC)NC(C(F)OC)=O 26900,C1(C(N2CCN(CC)CC2)=O)CNC(=O)CN1C(c1ccc[n+]([O-])c1)=O 26901,C1(CNC(CN(CCOC)C)=O)CC2CCC1N(C(C1CCC1C)=O)C2 26902,c1(C(C)=O)ccc(Cl)c(NC(C2COCCN2Cc2ccn(CCF)n2)=O)c1 26903,N1(C(C(C)CC2CCC2)=O)CC2(CCCN(C(=O)C=CC3(C)CCOCC3)C2)C1 26904,c1(OC(C)C(=O)NCC2(F)CCN(C(=O)CN3CCC3C)C2)ccc(F)nc1 26905,c1(OC)ccc(CC(=O)NC2(C)CN(C(=O)C(C)C3CCCO3)C2)cc1F 26906,C(=O)(CC(C)(C)C(F)F)NCC1(O)CCN(C(CC(C)(C)C)=O)C1 26907,C#Cc1ccc(C(=O)NC(CNC(c2cccn2C)=O)CC)o1 26908,c1(C(N2CC(NC(c3nc(CC)oc3C)=O)C(C(F)F)C2)=O)cc(C)nc(O)n1 26909,C1(C(=O)Nc2c(C)ncnc2)CC2CCC1N2C(C1CCC1C#N)=O 26910,N1(C(C(C=C)O)=O)CCC(CCCCNC(=O)C(n2ccc(C)n2)C)CC1 26911,S(=O)(=O)(c1cc(C(=O)NC2CC3(C2)CN(C(C24CC(C)(C2)C4)=O)C3)co1)NC 26912,Cc1cc(C(N2CCC(C)(NC(=O)CC3CCC(C)(C)O3)C2)=O)ccc1Cl 26913,c1(C(N(C(C)C)CCNC(C2CC3CCCCC23)=O)=O)cc2cc(Cl)cnc2o1 26914,CCC(C)(COC)C(=O)N1CCCC(CNC(=O)Cc2cc(C(F)(F)F)co2)CC1 26915,C(C(=O)NOCC(N1CCC(C(C)(C)C)C1)=O)=CC 26916,C1(C)(COC)CC(NC(c2ccc(N)cc2Cl)=O)CN1C(=O)C=C1CC1 26917,c1(NC(c2c(C)cccn2)C)nc(N(C)CC2CCC(=O)N2)c2ccsc2n1 26918,N1(C(c2cc(C)cnc2OC)C(=O)NCCCCCC)CCc2n[nH]cc2C1 26919,N1(c2c3ncn(C(C4CCC(C)C4)CO)c3ncn2)CC=C(c2cccs2)CC1 26920,CC1CN(CCNCC(c2ccc(OC(F)F)cc2)C)CC(C)O1 26921,C1(OC)(CNC(=O)CCC2CCC(C)O2)CN(C(=O)Cc2n[nH]c(C)n2)C1 26922,c1(SC)ncccc1C(=O)NC(=O)C(C)Cc1ccccc1.C12(C)CN(C1)C2 26923,c1(OC)cc2c(cc1C)CN(C(c1csc(C)n1)C(=O)NCCC1(C)CC1)CC2 26924,c1(C(=O)NC(C(C)NC(c2c(OC)c[nH]n2)=O)CO)cccc(CC(F)(F)F)c1 26925,Cc1cc(F)ccc1CNC(=O)NC1(CF)CCCC1 26926,CC1CCN(N2CCC(N)C2)CC1.C(=O)(CS(=O)(=O)N1CCN(C)CC1)NCC=O 26927,N1(C(CC(C=C)CC)=O)CCCCC2C1CCCN2C(=O)CC1(C)CCCC1 26928,C=CCC(C)(C)CC(=O)NCC1CC1CNC(c1nonc1CC)=O 26929,Cc1cc(C(=O)N(CCCNC(c2cnn(C3CC3)c2)=O)C)cn1C(C)C 26930,CC1CN(C(c2csc(S)n2)=O)CC1NC(c1ccncc1-n1cccn1)=O 26931,CCCC(C(=O)NCC(N1CCN(C(C)=O)CC1)=O)OCC1CCC1 26932,N1(S(Cc2c(C)nns2)(=O)=O)CC(=O)NC(C)C1 26933,c1(C(N2CC3C(C(=O)NCc4ncc(C)nc4)(C3)C2)=O)c(Cl)ccc(Br)c1F 26934,N1(C(CSCC=C)=O)CC(NC(=O)C(C)Cn2cccn2)C(C(F)F)C1 26935,C(=O)(C1=Cc2ccccc2C1C)NC(CCOC)CNC(c1nc(Cl)cs1)=O 26936,Cc1ccc(C=CC(N2CCCC(C(C)NC(=O)CC(F)(F)F)C2)=O)cc1Cl 26937,Cc1c(C(N2CC=CCC2C(=O)NOC2CCCC2)=O)nnn1C 26938,c1(C(=O)OC)nccnc1N1CCCC(C(C)NC(=O)CC2CC3CCC2O3)C1 26939,C1(CC)CN(C(c2ccnn2C2CCC2)=O)CCC1NC(=O)CC(C)(F)F 26940,N1(C(CCN(C(C(n2ccc(C)n2)C)=O)CCO)=O)CC2(C)COCC2(C)C1 26941,c1(C(=O)NCC(CNC(Cc2c(C)ccs2)=O)F)ccc2c(c1)NC(=O)C2(C)C 26942,C#Cc1cc(F)c(C(=O)N(C2CCC(NC(c3csc(C#N)c3)=O)C2)C)cc1F 26943,CCC(CC)(CC)C(=O)N1CCC(CC(=O)N(C2CCCC2(C)O)C)CC1 26944,c1(CNC(C2ON=C(CC)C2)=O)nn(C)c2c1CN(C(=O)C=C(C)C(F)F)CC2 26945,C1(NCc2nc(SC)nc(O)c2)CCC2(CC1)CC(O)C2 26946,CCC(C(=O)NCCCN(C(=O)C(C)NC(N)=O)CC)N(C)C 26947,C(CCC(C(=O)N(C)Cc1nncn1C)NC(c1csnc1Cl)=O)OC 26948,c1(NC(C(C2CCSC2)N(CCC(=O)OCC)C)=O)ccccc1C 26949,Cc1ccc(C(=O)NCCC(O)CNC(C2CC(O)C2)=O)c(N)n1 26950,c1(CCC(=O)NC2CC(C(=O)NCC3(SCC)CC3)C2)nc(O)n[nH]1 26951,N1(C(c2ccc(C)nc2)=O)CC2CCN(C(=O)COCP(C)(C)=O)C2C1C 26952,C(CCCC(=O)NC1CC1)N(C)CCNC(CCF)C(=O)N(C)C.C(=O)O 26953,N1(c2ccnc(C(=O)OCC)n2)CCC(C)C(NC(=O)C(F)C(C)C)C1C 26954,C1(CC(N2CCC(NC(C)=O)C2)=O)CCN(C(=O)Cc2cnnn2C)CC1 26955,c1(COC2CCCN(C(CNC=O)=O)C2)cccc2cncn12 26956,N1(C(C2C(=C)C2)=O)CC=C(C(=O)NCC2Cc3nccn3C2)CC1 26957,c1(C(=O)NC(C(=O)NC(C2CCOCC2)C)Cn2cccn2)cccc(CO)n1 26958,c12cc(n[nH]1)C(=O)NC2.N1(C(C(C)C2CCC2)=O)CCCC1c1ncc[nH]1 26959,Cc1nc(C=CC(=O)NC2(CCNC(C3(CC(C)C)CCC3)=O)CC2)cs1 26960,C1(C)(C(=O)NCC(CN(C)C(c2csc(-c3ccco3)n2)=O)O)C(C)(C)C1(C)C 26961,C1(C(=O)NCCC2N(C(c3cn(CC)nc3)=O)CCCC2)CC2CCCCCC12 26962,C1(C)(C(=O)OC)CCN1C(=O)CCOC1CN(C(=O)C(=O)C2CC2)C1 26963,C1(C(=O)OCC)(NCCc2ccn(C)n2)CC2CC1C1CC(C)CC21 26964,N1(C(c2scc(NC(C)=O)n2)=O)CC2CN(C(c3ccc(C)nc3)=O)C2C1 26965,C1(NC(C(C)(C)OC(C)=O)=O)CCCC1(C)NC(=O)C=C(C)Cl 26966,C1(c2nnnn2C2CCOC2)(Nc2ccc(NC(C)=O)cc2)CCCC2(CC2)C1 26967,C1(C(N2C3CC(NC(C4(C#C)CCC4)=O)CC2CC3)=O)CCc2c(n[nH]c2C)C1 26968,N1(C(=O)OC(C)(C)C)CCC(NCC2CCN(CCc3ccccc3)C2)C(O)C1 26969,CCCCCCCC(=O)NC(CC)CCC(=O)N(C)CC1CCOCC1 26970,C1(C(N2CCC(CCC(=O)NC(c3nccs3)CC)C2)=O)CCCC1C1CC1 26971,CCCCC(CC)C(=O)N1CCN(C(=O)Cc2ccnn2C)CCC1C 26972,N1(C(C(C)NC(CC)=O)=O)CCC12CN(C(=O)C(C)(C)c1cc[nH]n1)C2 26973,O=C1Cc2c(C(N3CC4(CCN(C(C5C6CCC(=O)C56)=O)C4)C3)=O)cccc2N1 26974,C1(NC(C)=O)CCN(Cc2ccc(C#N)s2)CC1C 26975,c1(CC)n[nH]cc1C(N1CCCC1CCNC(=O)CNC(C1CCC1)=O)=O 26976,C1(NC(C(CSC)C)=O)CCN(C(c2cc[nH]c(=N)n2)=O)C1C 26977,c1(C(=O)NC2CC(C)(C)N(C(C3CNC(=O)N3)=O)C2)cccc2nc(CO)[nH]c12 26978,N1(C(CC2C(C)CCC2)=O)CCCC(C)(CNC(c2scnc2C(C)(C)C)=O)C1 26979,c1(C(N2CCC(NC(C3CCCCS3)=O)CC2)=O)ccc([N+](=O)[O-])cc1O 26980,N1(C(c2c(C)n(C)nn2)=O)CC(F)(F)CC1CCNC(=O)C1=C(Cl)CC1 26981,c1(CSC)cc(C(=O)NCC2CC(OC)CN2C(=O)C2=COCCO2)ccc1F 26982,N1(C(c2c(C)nc(CC(C)C)o2)=O)CC2CCC1CN2C(=O)CN1CCC1C 26983,C1(NC(=O)CCN2CCCC2)CN(C(c2cnc(O)o2)=O)C2(CCOC2)C1 26984,N1(C(CC2CC(SC)C2)=O)CC2(NC(=O)CCc3ccnc(Cl)c3)CC1C2 26985,C1(NC(C(CC)N(C)C)=O)CC2CCC1C1CN(C(c3ccc(=O)oc3)=O)CC21 26986,n1(CCc2onc(-c3ccc4ccn(C)c4c3)n2)cnc2ccccc2c1=O 26987,c1(NC2CCCC(NC(=O)CCCc3cccnc3)C2)ncnc2c1CCO2 26988,C1(C(=O)OC)(C(=O)NCC(O)CN(C)C(c2cc(O)ncn2)=O)CCCCO1 26989,C(=O)(C(C)(C)CS(C)(=O)=O)NC1CC(C)CN(C(=O)Cn2nc(O)ccc2=O)C1 26990,C(N(C)N1CCC(C)(CC(=O)OC)CC1)c1cccc(OCC)c1 26991,N1(C(CCC2CCC(=O)N2)=O)CCCC(F)(C(=O)NC2CN(CC(F)F)C2)C1 26992,N(C1CCOc2ccc(F)cc21)C(c1ccc(SC(F)(F)F)cc1)C(=O)OC 26993,NS(=O)(=O)c1ccc(C(N2CCC(CNC(=O)Cc3cc[nH]n3)C23CC3)=O)o1 26994,c1(C(=O)NCC(CCNC(CCCC(C)=O)=O)(C)C)cc2c([nH]1)CCCC2 26995,c1(C(C(=O)NC2CC(F)(F)C2)N(CC(=O)NCCC)C)nc(Cl)cc(Cl)c1C 26996,c1(OCCOC)ncccc1C(=O)NC1CCC(NC(=O)C(F)(F)CO)CC1 26997,N1(C(c2ccco2)=O)CCC2(C(N3CCN(c4ncccc4Cl)CC3)=O)CC2C1 26998,N1(C(COC(CC)C)=O)CCC(CNC(=O)Cc2cnsc2)C(CC)C1 26999,c1(OC)cc(Br)c2c(c1)CCN(C(=O)C(=O)NCC1(OC(C)C)CCOCC1)C2 27000,N1(C(c2cccc(COC)c2)=O)CCC2(CCCN2C(c2ccc(Cl)o2)=O)C1 27001,N1(C(c2c(CC)occ2)=O)CC(NC(C23CC(CC)(CO2)C3)=O)C(C(F)(F)F)C1 27002,CCCC(C)(CC)C(=O)NC1CN(C(c2cc(C3(C)CC3)n[nH]2)=O)CC1F 27003,Cc1cc(N)c(C(=O)NCC#CCNC(=O)C(C)(O)c2ccccc2)cc1C 27004,C(CN(C(=O)Cn1cnnn1)C)(CO)(CO)NC(C(N1C(=O)CCC1=O)CC)=O 27005,N1(C(c2[nH]cc(C#N)c2)=O)CCC(CCNC(=O)CC2OCCCO2)C(F)(F)C1 27006,S(=O)(=O)(c1ccc(Br)cc1NC(CO)CC#CC)NCCC=C=C 27007,C1(CC(C)NC(C2C(OCC)C2C)=O)CCN(C(=O)C(C)OCC)CC1 27008,C=CCC(CC=C)C(=O)N(C1CN(C(C2(COC)CC=CC2)=O)CC1F)C 27009,c1(OCC)ccccc1C(=O)NC1N(C(COCC=C(C)C(F)CBr)=O)CCC1 27010,CCCCCCC(CC)NC(C1CCCCCN1C(c1n[nH]c(C)c1O)=O)=O 27011,N1(C(C2N(C)CC(C)(C)C2)=O)CC=C(CC(=O)NCC23CCCC2C3)CC1 27012,N1(C(CC(CC)C2CC2)=O)CCC2C(C1)CN2C(c1csc(Br)n1)=O 27013,C(C1=NOC2OCCC12)NCC(C(=O)N(c1ccccc1)C(C)C)C 27014,CC1CCC(=CC(=O)NC(C)(C(=O)NC(c2cscn2)C)C2CCC2)CC1 27015,CCC(CC(=O)NCC(C)(C)CCNC(=O)C(C)COC)C(C)C 27016,C1(NC(CC2C(C)=NNC2=O)=O)C2CCCN(C(C3CC3C)=O)C2C1(C)C 27017,c1(C2CN2)ccc(N2CCCCC2)cc1.CC1CC(CS(=O)(=O)N(C)C)CN1 27018,N1(c2nnc(OC)c(OC)c2)CCC2CN(C(C)=O)C2C1 27019,N1(C(CN2CCN(CCCC=C)CC2=O)=O)CCn2c(C)nnc2C1 27020,C1(C)(NC(C2(C)N(C(CCSCC)=O)CC=C2)=O)CCC(C)=C(C)C1 27021,C1(C(=O)NC(C(=O)NC2CC(C(=O)OC)C2)C)CCC2(CCC2)C1 27022,C(=O)(C1=CCCC1P(C)(C)=O)NCCN(C(CC(C=C)(C)C)=O)CC(C)O 27023,C(=O)(C(Cc1cn[nH]c1)NC(=O)Cc1cnns1)NCCC(C)SC 27024,C(C)(C(N)CC(=O)N1CCCC1CC(c1cccs1)O)OCC 27025,N1(C(CCN(CCC)C)=O)CC2(CCC(NC(=O)CCc3ccncn3)CC2)C1 27026,N1(C(C(=O)N(CC(C)NC(CSCC)=O)C)CC)C(=O)c2ccccc2C1=O 27027,c1(C(C)=O)ccc(CC(=O)NCC(C)(C)NC(=O)CC2CCC3CC23)cn1 27028,C(=O)(C1=NOC2(CCC2)C1)N(CC(CC)NC(c1cc(C#N)oc1C)=O)C 27029,CC(C)(O)CC(=O)NCC1(C(=O)NCc2ccc(C3CC3)o2)CCCCC1 27030,CC1(C)CC(C#N)(CNC(C2CCCCCN2C(C2CCC(O)CC2)=O)=O)C1 27031,CS(=O)(=O)c1ccc(C(=O)NC2CCN(C(=O)C(F)C3CNC3)CC2)cc1 27032,C1(CNC(c2scc(C)c2)=O)CN(C(=O)CC2CCCC23CC3)CCO1 27033,c1(CC(N2CCN(C(c3ccnc(C)n3)=O)C(CO)C2)=O)coc2ccccc12 27034,c1(C(=O)NCC(C)(CC)NC(C(F)=CCC)=O)cc(OC)cc(OC(F)F)c1 27035,CC1(C)CC(c2nnnn2CCCF)(NCCSc2ccc(Br)cc2)C1 27036,C(=O)(C1=C(Cl)CCOC1)NC(COCC)C(=O)NC1CC1(C)C(F)F 27037,c1(OCC)ncc(C(=O)NC(C)(C)CCCNC(=O)Cc2ccno2)cc1Cl 27038,C1(NC(C(CCC)O)=O)CCN(C(C2CSC2)=O)CC1C 27039,c1(C(=O)NC2C(NC(CC(C=C)C)=O)CCC2)ccc(C)c(Br)c1N 27040,c1(C(=O)NCCOC(CNC(C(C(C)O)C)=O)(C)C)cc2n(c1)CCCC2 27041,c1(C(=O)NC(C)CCc2cccn2C)cc2c(cnn2C)nc1C(F)F 27042,c1(OCC(=O)NCC2CCCO2)cccc(OC(F)F)c1.C12CC(C1)CNC2=O 27043,N1(C(C(C)NC(N)=O)=O)CCCC(C)(NC(C2CCC(=O)NC2)=O)C1 27044,N1(C(c2nc(CC)oc2)=O)CC2CCC2(C(=O)NC(CO)CC(C)C)C1 27045,n1(C2(C(=O)NC(C)C(C)NC(=O)Cc3cc(C4CC4)on3)CC2)cc(Br)cn1 27046,c1(CC(=O)NC2CCCC(NC(C(C=C)O)=O)C2)cc(F)ccc1Cl 27047,N1(C(c2c(C)cco2)=O)CC2CCC1C1CN(C(c3occc3F)=O)CC21 27048,c1(CC(=O)NCC(O)CNC(C23CCC(C2)C3)=O)cccc(Cl)c1 27049,C1(C(=O)NC(C#C)CC2CCCC2)C(CC)CCN1C(c1csc(CC)n1)=O 27050,N1(C(c2cccc(F)n2)=O)CCCC(C2CCN(c3ncnc(Cl)c3F)C2)C1 27051,N1(C(CCCOc2ccc(C(C)=O)cc2)=O)CCC(C2(C(=O)O)CC2)CC1 27052,C1(COC)CCC(C(N(C2(C(=O)Nc3ccsn3)CC2)C)=O)C1 27053,Cn1c(C(N2CCC(O)(CNC(C3(C)CCNC(=O)C3)=O)C2)=O)ccc1C#N 27054,C1(OCC#C)CCCN(C(C23CC(NC(=O)C(Cl)Cl)(C2)C3)=O)C1 27055,N1(C(c2nc(C(C)OC)sc2)=O)CCCC(N(C(=O)CC2CCC(=O)N2)C)C1 27056,C1(C(N2C(CNC(=O)C=C3CCC3)CC2)=O)CC12CCC1(CC1)CC2 27057,c1(C(=O)NCC(CC)NC(=O)COCC2CCOC2)ccnc2c(Br)cccc12 27058,C1(NC(c2cncc(C)c2)=O)COC2(CCN(C(=O)CC34CCCC3C4)CC2)C1 27059,C1(C2CC2)(C(=O)NC2CCC(NC(CCC(=O)OC)=O)C2)CCOCC1 27060,C(=O)(C1CCc2nccn21)N1C2(C(N3CC(C(=O)OC)(CC)C3)=O)CC2CC1 27061,c1(OCC)cncc(N2CCCC2Cc2ccc(C)cc2)n1 27062,c1(C(=O)NCCC(C)Nc2ncncc2Cl)ccc2scnc2c1 27063,c1(C(=O)NC2(CCC(=O)NCCCCC(=O)NC)CCC2)cc(C)nc(C)c1 27064,C(=O)(C(C)C(=O)OCCC(C)C)NC(CN(C(COC)=O)C)C 27065,c1(CNC2CN(C(=O)OC(C)(C)C)C2(C)C)c(F)cc(Cl)cc1Cl 27066,c1(C(=O)NCCC2CCN(C(c3cnc(C(=O)OC)s3)=O)C2)nnn(C)c1C 27067,N(C(=NCCF)NCC1(O)CCS(=O)(=O)C1)CC1CC(OC)CN1C 27068,N1(C(Cn2ncc(C)c2)=O)CC(C)(CNC(C2(F)CC=CC2)=O)CC1(C)C 27069,C1(CNC(=O)NCC(C(=O)OCC)(C)O)OC(C)(C)OC1C(=O)O 27070,c1(C(=O)NCC(C)(CNC(=O)CSc2nnnn2C)OC)ccc2n[nH]cc2n1 27071,C(=O)(C1=CSCCO1)NC1C(CNC(CC2C(C)=NNC2=O)=O)CCC1 27072,C(=O)C(=O)CC(C)CC.c1(C(=O)NCCC=CCCC)ncoc1C 27073,Cc1c(C(N2CC3C(CN(C(=O)CCCC4CCC4)C)C3C2)=O)cnn1C(C)C 27074,N1(S(CC)(=O)=O)CCCC1C(=O)NCC(c1ccccc1)NC(=O)C1=CCC1 27075,N1(C(CCP(C)(C)=O)=O)C2CCC1CC(NC(C1CCOC3(CCC3)C1)=O)C2 27076,CC1CCC(CO)N(C(C2C3CC4C(C3NC(c3cc(O)ncn3)=O)C24)=O)C1 27077,N(C(=NCCc1ccc(Br)cc1Cl)NC1CC1)CC1CCN(C)C1=O 27078,CC1C2CCC(C2)C1C(=O)N(C)CC1CCC(CNC(=O)Cc2nc[nH]n2)CC1 27079,N=c1nc(O)c(CC(=O)NCC2CC2CNC(=O)C(O)CN(C)C)c[nH]1 27080,CCCS(=O)(=O)C(C)C(=O)N(CCCNC(=O)COCc1nccn1C)C(C)C 27081,C1(NC(c2c(C)cns2)=O)CC2CC1CN(C(=O)C(C1CCCCCC1)O)C2 27082,CCC(F)C(=O)NCCN(C(=O)CC1CC=CC1)C 27083,c1(CNC(c2c(-n3cc(CC(C(C)C)O)nn3)cccc2)=O)cccc(F)c1F 27084,N1(C(C(c2cccc(F)c2)C)=O)CC(CNC(c2n[nH]c(O)n2)=O)C(C)C1 27085,N1(C(C2C(C=C)C2)=O)CCCN(C(c2ccnn2CCOC)=O)CC1CO 27086,C(=O)(C1=CC2(CCN(C(C34C=CC(CC3)C4)=O)C2)C1)N(CC(F)Cl)C 27087,C1(CNC(CC(=O)NCC)=O)N(C(=O)CC2CC(C)(C)C(=O)N2)CCC1(C)C 27088,N1(CC(N2CC(C)(NC(=O)Cc3ccc(C#N)cc3)C2)=O)CCn2ccnc2C1 27089,C=CCCC(C(=O)NCC(CC)C(C)(F)F)NC(C1CCC(OC)CC1)=O 27090,c1(C(=O)NCC(C)NC(=O)CN(C)CCO)cc(Cl)c2n[nH]cc2c1 27091,Cc1cc(C(=O)NCCC2CCC(NC(=O)CC(C)C)C2)c(N)c(Cl)n1 27092,c1(NC(=O)C=CC2CC2)cccc(CNC(c2nc(C(F)(F)F)cs2)=O)c1 27093,C1(CN(C)C(c2cn(C)nn2)=O)CCC(NC(=O)CC2CCCC(=O)N2)CC1 27094,c1(C(=O)NCCC(C)NC(C2(CC)CCCO2)=O)ccc(CN2CCCC2)cc1 27095,C1(CCOC)CN(C(c2ccc(C(O)CF)cc2)=O)CCN1C(C1CC1F)=O 27096,c1(C(=O)NC(CC)CN(C(=O)CC2CCOC2)C)ccnn1C(F)F 27097,C(C)(CCCC(=O)N1CCC(CCO)CC1)NC(C(C)OCCCC)=O 27098,C1(C(=O)NC2CON(CC)C2=O)CN(C(c2ccc(C)nc2O)=O)CC1(F)F 27099,N1(C(c2cc(CCC)on2)=O)CC2CCC2(CC(=O)N(CCC(=O)NC)CC)C1 27100,c1(CCC)onc(C)c1C(=O)NCC1(C)CCN(C(C2(C#N)CCCO2)=O)C1 27101,C=CC1(C(=O)NC2CN(C)CCC2O)CCN(C(=O)C2=NOC(C)C2)CC1 27102,C1(NC(c2n(CC=C)ccc2)=O)CN(C(c2cccc(C)c2)=O)CC(C)(C)C1 27103,CC1CC(C)CC2(C1)NC(=O)N(CC(=O)NC1CC3CC1C(O)C3O)C2=O 27104,Cn1cc(C(=O)NCC2CCCC(NC(c3sccc3C(F)F)=O)C2)ccc1=O 27105,c1(-c2cccc(C3C(C(N4CCC5(CCCC5)C4)=O)C3)c2)cccc2c[nH]nc12 27106,CN=c1[nH]c(=NCCc2cc(O)ncn2)[nH]c(=NCC(C(C)C)OC)[nH]1 27107,c1(C(=O)NCC2C(NC(c3cc(CC)oc3C)=O)CCC2)ccc(C)cc1OC 27108,N1(Cc2c(=N)cc[nH]c2)CCCC(C(N2CC3CCCC23)=O)CC1 27109,Cc1cccn2ncc(C(N3CC(O)(CN(C)C(C4CNC(=O)N4C)=O)C3)=O)c12 27110,C1(C(=O)NCC2CC(NC(C(C)OC)=O)C2)CC2CCC1O2 27111,N1(C(CCC#CC)=O)CC(NC(=O)C(C)(O)c2ccccc2)CC2(CC2)C1 27112,C1(CC(=O)NC2(CN(C(=O)CCCc3ccsc3)C)CC2)CCC2CC2C1 27113,CN1CC(F)CC1C(=O)NCC1CCC(NC(C2CC2CC(C)(C)C)=O)C1 27114,C1(CNC(CC(C)C#N)=O)CC2(C1)CN(C(=O)Cc1ccoc1)C2 27115,C1(CCNC(C2C(OCC)C2)=O)CCCN1C(=O)CSC(F)F 27116,c1(C(=O)NCC2CC(NC(c3c(C(C)C)ocn3)=O)C2)ccc2c(c1)CCC=C2 27117,C1(C(=O)NCCCCN(C(C2(COC)CC=CC2)=O)C)CCC(C)(C)CO1 27118,C1(CC(=O)N(CC(C)(C)CNC(=O)CCc2ncnn2C)C)CCCCC(=O)N1 27119,c1(C(=O)NC2CCN(C(c3sccc3Cl)=O)C2)nnn2c1C(=O)NCC2 27120,C(=O)(C1=NOCC1)N1CCC(CN(C(C(CC)OC)=O)Cc2ccccc2C)C1 27121,C(C(CC(C)C)C(=O)NCC(CC(C)C)OC)NC(CC(C=C)(C)O)=O 27122,c1(N(C(=O)NC)CC)ccc(C(=O)NC(c2cccnc2)C2CCOC2)cc1 27123,C1(C(=O)NC(C)CC2CN(C(=O)CCc3cnoc3)C2)CCc2nncn2C1 27124,C1(C(=O)Cl)(NC(c2cccnc2C2CC2)=O)CCOCC1.N12CCCC(C1)C2 27125,c1(NC(=O)NCc2c(CCC)cccc2)cc(C(C)C)cc([N+](=O)[O-])c1 27126,C(=O)(C(F)CC(C)(C)C)NCCN(CCC)C(c1ncccc1N)=O 27127,Cn1nc(Br)cc1C(N1CCC(CC#N)CC1)C(=O)NC1CC(F)(F)C1 27128,N1(C(C(CC(CC)C)C)=O)CC(C)CN(C(c2cccc(OC)c2N)=O)CC1C 27129,C12(CNC(C(CC3CC3)NC(=O)CC34CCCC3C4)=O)CCC(CC1)O2 27130,Cc1ccc(C(=O)NC2CC(CC(N3CCOC(C4CC4)C3)=O)C2)c(F)c1 27131,N1(C(C(C=C)OC)=O)CC2(C=C(C(=O)N3CCCC3C(=O)NC)CO2)C1 27132,N1(C(C(C(=O)NC)(C)C)=O)CC(C(=O)N(C)CCc2nccs2)CCC1(C)C 27133,C(=O)(CC(CC)C(C)(C)C)N(C1CCN(C(=O)CCCNC(C)=O)CC1)CCC 27134,C(CC(C)(C)C(=O)NC(CNC(=O)COCCF)C1CCC1)OC 27135,S(=O)(=O)(c1cc(F)cc(F)c1)N1C2CC(N(CCC#N)C)C(C2)C1 27136,C(=O)(CC1OCCc2ccsc21)N1CC(NC(C(CC#C)CC#C)=O)C(C)(C)C1 27137,C(C1c2ccccc2CC1C)NC(N1CCC(c2ccc(C)cc2)C1)=O 27138,c1(OC)cc(CN=c2cc(CC(=O)OC)nc(C3CC3)[nH]2)c(F)c(F)c1F 27139,C1(NC(c2ccn(C(F)F)n2)=O)CC(O)CN1CC1CCCN1C(C1CCC1)=O 27140,n1(CC(=O)NCC2COCCN(C(c3csnn3)=O)C2)nc2c(n1)CCCC2 27141,C1(CCNC(c2ccc(N(C)C)cc2)=O)CN(C(C2(F)CCC2)=O)CCCO1 27142,c1(N2CCC(N(C(C3C(C)C3)=O)C)C2)nc(Cl)ncc1C1CC1 27143,c1(C(N2CC(=C(CNC(=O)Cn3c(O)nnc3O)F)C2)=O)n[nH]cc1[N+](=O)[O-] 27144,CN1CC2CCC(C1)N2C(C1CC12CN(C(C1CC1c1ccc(O)cc1)=O)C2)=O 27145,CC1(NC(=O)CNc2ncccn2)CC(NCC2CC2)C1 27146,N1(C(C(C)O)=O)CCN(C(c2sc(Br)nc2Br)=O)CC1CO 27147,C12CC(F)(F)CN1C(=O)NC2.C(c1ccccc1)=C(CC)C(=O)OC(C)(C)C 27148,N1(Cc2c(C)cccc2Br)CCC2CN(C(=O)C(C)n3ccnc3)CCC12 27149,Cn1c(=O)n(C)c2cc(CS(=O)CC3CC4(CCC(C(=O)O)CC4)C3)ccc12 27150,C(CN=c1cc[nH]cc1S(=O)(=O)NCCCCF)c1c(C)c(Cl)c(Cl)cc1 27151,c1(C(=O)NCC(C2(O)CCN(C(c3cc(Cl)n(C)n3)=O)C2)C)ccc([N+](=O)[O-])[nH]1 27152,c1(C(=O)NCC=CCNC(CN2CCC(C)C2)=O)cc(Br)cnc1NC1CC1 27153,N1(C(C2C(C)C2)=O)CCOCCC1C(=O)Nc1cnc(C(C)C)nc1 27154,CCC(F)(F)CC(=O)N1CCC(C)C(NC(=O)Cn2cnc(Br)c2)C1 27155,C(CNC(=O)Cn1cc(N)cn1)(C(C)(C)C)NC(C1(CC=C)CCC1)=O 27156,c1(C(N(C2CCCCN(C(C3CC3C(N)=O)=O)C2)C)=O)cc2cn[nH]c2cn1 27157,C1(NC(C2CCC(CC)O2)=O)CCN(C(c2cc(C)cc(Cl)n2)=O)CCC1CO 27158,C1(CNC(C2(CCCC)CCCC2)=O)CCN(C(=O)CCc2nc[nH]n2)CC1O 27159,N1(C(Cn2cc(C(=O)OCC)nn2)=O)CCN(C(=O)CSCC)C(C(C)(C)C)C1 27160,C(CNC(C1CC1c1cccc(Cl)c1)=O)(C(C)(C)C)NC(C12CC(C)C1C2)=O 27161,C1(CC(C)NC(C2(CN(C)C)CC2)=O)CN(C(C2CCC2)=O)C1 27162,N1(C(CCn2cc(CNS(CC)(=O)=O)nn2)=O)CCCC(CC(=O)OC)(OC)C1 27163,C1(N(C)C)CCN(C(=O)CCNOCc2ccccc2)C(C)(C)C1 27164,N1(CC(N)=O)CCCC(C2CCN(C(C3CC34CCOC4)=O)CC2)C1 27165,N1(C(CCn2c(C)ncc2)=O)CC2CC(NC(C3CCC4(CCC4)O3)=O)C(C2)C1 27166,N1(C(CCSC)=O)CCOC(C(C)NC(c2cccc(N(C)C)c2)=O)C1 27167,Cc1ccc(CC(C)C(=O)N2CCC2CNC(=O)Cc2ccc(Cl)cn2)cc1 27168,N1(C(CSCCC#N)=O)CC2CC(NC(=O)Cc3csnn3)CC2C1 27169,C(CC(C)(C)C)(C(=O)NC1CCC1NC(c1ccc(F)c(CC=C(C)C)c1)=O)OC 27170,O=C1CCN(CC(=O)NCCNC(=O)CC2CC=CCC2)CC1 27171,C(=O)(C(C)C(O)CC)NC(CC=C)C(=O)Nc1ccc(CO)cc1O 27172,C(C(C)C(=O)NOCC1CCOCC1)NC(C(COC)(C)OC)=O 27173,CC(=O)CCCC(=O)NCCCN(C(C1CC(C)(C)CCO1)=O)C1CC1 27174,N1(C(c2ccn3c2CCCC3)=O)CC2CCCC(O)C2C1 27175,N1(C(C(C2CC2)SC)=O)CCC(O)(C(C)NC(C2CCCN2C(=O)C2CC2)=O)C1 27176,c1(C(=O)NC2C3(CC(NC(C4=NOC(C)C4)=O)C3)C2)cc2cc(Cl)ccc2o1 27177,c1(C(N(C)CC2CCCN(C(C(C(C)O)(F)F)=O)C2)=O)c(F)cc(F)c(F)c1F 27178,c1(SC)cc(C(=O)N(CCC(C(C)(C)C)NC(=O)C=CCO)C)ccc1N 27179,C(=O)(C1=CC2(CCOC2)C1)NC(CC(=O)NCc1cccnc1O)C(F)F 27180,c1(OC)cnc(C(N2CCC(N(C(=O)C=Cc3cncs3)C)C2)=O)nc1 27181,Cc1c(C(=O)NCC(C)N(C)C(C2CCC(=O)N(C)C2)=O)nn2ccccc12 27182,N1(C(CCC(C)(F)F)=O)CC(NC(=O)CS(=O)(=O)C2CC2)CC12CCC2 27183,n1(CC(=O)NCC2CC2CNC(C2CCC(CCO)CC2)=O)ccc(O)nc1=O 27184,N1(C(c2c(C)cc(C)s2)=O)CCC(CO)C(NC(=O)Cc2cccnc2C)C1 27185,C1(CC(=O)NCCN(C)C(c2ccnc3ncnn23)=O)CCCCCC1(F)F 27186,c1(C(N(C2CCCN(C(c3csc(F)c3)=O)CC2)C)=O)cccn(C)c1=O 27187,c1(OC)cccc(C(=O)NCC2CC(NC(=O)CCCC(N)=O)C2)c1O 27188,N1(C(C2C(CC)CCCC2)=O)CCC(COC)(NC(=O)CCC2(C)CC2)CC1 27189,C1(NC(c2c[nH]nc2CCNC(c2cccc[n+]2[O-])=O)=O)CC1C1CCC1 27190,CCC(C(=O)NCC12CC(NC(=O)C(F)OC(F)(F)F)(C1)C2)n1ccnc1 27191,c1(NC2CCC(NC(C3C(=C)CC3)=O)CC2)cc(OC)nc(-c2cccnc2)n1 27192,Cc1cc(C)c(CNCC2COCCN2c2ncc3ccsc3n2)c(C)c1 27193,Cc1ccc(C(=O)N(CCCNC(C2C3CCCCCC23)=O)C)c(O)c1C 27194,c1(CC)nc(NC2CN(C(=O)CC3CCCC34CC4)CC2C)c(C#N)cc1C 27195,C1(C(N2CC(NC(=O)CCOc3cccc(Cl)c3)C(F)C2)=O)CCCC2(CC2)C1 27196,C1(NC(CCSCCC)=O)CC2CCC1CC2NC(c1csc2nccn12)=O 27197,c1(C(=O)OC)oc2cccnc2c1NC(C1(CNCc2cccc(F)c2)CC1)=O 27198,N1(c2ccnc(OC)n2)CC2(CCCN2C(c2ccsc2C)=O)C1 27199,C1(C(N2C(C(=O)OC)CC2)=O)CCCN1C(c1ccc(Cl)o1)=O 27200,c1(C(N2CC(NC(C3CCOC(=O)N3)=O)CC(C)C2)=O)ccc2ccn(C)c2c1 27201,C1(F)(C(=O)NCCc2onc(C)n2)CCCN(C(=O)C=C2CCC2)C1 27202,Cc1c(O)ccc(C(N2CCCC(C(C)NC(C3(CF)CCC3)=O)C2)=O)c1C 27203,C1(NC(CCc2cc(C)on2)=O)CC2CCC(C1)N2C(C1COC(=O)O1)=O 27204,C(=O)(C1=CCCCO1)N1CC(n2cc(CNC(C3(COC)CCCO3)=O)nn2)C1 27205,C(=O)(CC1OCc2ccccc21)NC(C1CCCCC1)CNC(=O)C#CC1CC1 27206,C1(C(N2CC3=C(CN(C(CC(=O)OC)=O)C3)C2)=O)C2Cc3c(Cl)cccc3C12 27207,C1(C)(C(NOC(CC)C)=O)CN(C(=O)C=Cc2cnn(C)c2)C(C)(C)C1 27208,CC1CN(C(=O)Cc2cccc(F)c2)CCC1C(=O)NC1CC(=O)N(O)C1 27209,CC1CC(N(C)C(C2CSCCN2C(=O)CCN2CCOCC2)=O)CC(C)C1 27210,N1(C(C(COC)NC(c2[nH]nnc2C)=O)=O)CCN2CC(F)CC2C1 27211,c1(C(N(C2CN(C(C3CC(CF)C3)=O)CC2F)C)=O)cnc2c(C#N)cnn2c1 27212,CC1(C)CC(c2nn[nH]n2)CN(S(=O)(=O)CC2(C)CCCC2)C1 27213,Cc1cccc(CNC(C2CC2c2ccccc2-c2cncn2C)=O)n1 27214,c1(CN2CC3(C(C(N(C(C)(C)C)CCN)=O)C3)C2)cc(Br)c(F)cc1Cl 27215,C1(C(=O)NCC2CCCN(C(C3OCCN(C)C3)=O)C2)CCC(=O)N(C)C1 27216,c1(C(=O)NCCCCCNC(CC(CC)C2CC2)=O)cc2ccccc2n1CC 27217,C(C(O)CN=c1[nH]c(SC)nc(C)c1C)NC(c1ccc(OC)c([N+](=O)[O-])c1)=O 27218,c1(CN2CCC(CSC)C2)nnc(NC2CCCCC2)n1C1CCCC1 27219,C1(NC(CCC(=C)Cl)=O)CCCC12CN(C(C1C3CC4C(C3=O)C14)=O)C2 27220,C(CC(C(=O)NCC=CBr)NC(=O)COCC(C)C)=CC 27221,N1(C(c2cc(C(C)=O)c(C)o2)=O)CCC2CN(C(C3CC(OC)C3)=O)CCC2C1 27222,N1(C(C(CCOC)(C)C)=O)CCCC(C2CN(C(C3(S(C)(=O)=O)CCC3)=O)C2)C1 27223,c1(C(=O)NC(C(=O)N(C)CCn2ccnc2)Cc2cc[nH]n2)cn2ccccc2n1 27224,C12(CC(=O)NCC#CCOC)CCC1CN(C(c1csc(C)c1)=O)C2 27225,c1(C(=O)NCCCN(C(C(C)NS(CCC)(=O)=O)=O)C)cccc2c1OCC2C 27226,C1(C(=O)NCCC(C)(C)NC(c2c(C(C)(C)C)noc2)=O)C2CCCC(F)(F)C12 27227,CCCCCC(O)C(=O)NCC1CN(C(C2COCCN2C)=O)C1 27228,N1(C(C(CCNC(CCN(CCC)C)=O)O)=O)CCCCC(C)(F)C1 27229,c1(C(=O)NCCCN2CCC(NC(c3cc[nH]n3)=O)C2)cc(F)cc([N+](=O)[O-])c1 27230,C12(CNC(c3c(OC)c[nH]n3)=O)CCC1CCN2C(c1cnco1)=O 27231,C1(NC(CCCOCC)=O)CN(C(=O)CN2CCN(C)C(=O)C2)CCC1C 27232,CC1C(NC(=O)COCCCF)CCN1C(=O)CCCCN1CCOCC1 27233,CCC(CNC(C1CC(OC)CN1C(=O)CSc1ccccn1)=O)CC(C)C 27234,N1(C(C2N(C(CC3CC(=C)C3)=O)CCC2CC)=O)CC(C2CCCC2)C1 27235,C(C)(C)(CC(C)NC(=O)C(F)C1CC(NC(=O)CCN2CCCC2=O)C1)OC 27236,c1(C(=O)NCCN(C(C2(CC)CCOC2)=O)C)ccc(C(C)C)nc1O 27237,c1(CNC(C2(C)C(C)(C)C2)=O)nnc2n1CCN(C(c1ccc(Cl)c(N)c1)=O)C2 27238,Cc1sc(C(=O)NCC23CC2CN(C(=O)CN(C)C(C)C)C3)nc1O 27239,c1(C(=O)NCCN(C)C(C2CCCOCC2)=O)ccc2c(c1)CCCC(=O)N2 27240,C1(CNC(=O)NC(c2ncccc2Br)(C)C)CCCOC1c1cn[nH]c1 27241,N1(C(CC=C=C)=O)CCCC(NC(c2coc(Cl)n2)=O)CCC1 27242,Cc1cc(O)cc2c1CN(C1CC3CC1N(C(c1ccoc1I)=O)C3)CC2 27243,c1(CCC(=O)N(CC(C)NC(c2ncccn2)=O)C)nc2cc(Cl)ccc2s1 27244,n1(CCC)cc(C(=O)NC2CC(N(C(=O)Cc3cccn3C)C)C2)c(C)n1 27245,C1(C#N)(COC)CCN(C(c2cc(C3CCCN3S(C)(=O)=O)[nH]n2)=O)CC1 27246,c1(-c2n(C)cnc2)cccc2c1CN(N1CCC(c3ncc(CO)[nH]3)CC1)C2 27247,CC(C(CO)NC(c1cnc(C2CC2)[nH]1)=O)NC(=O)C(c1cccn1C)=O 27248,c1(C(N(CCNC(c2n(CC)c(O)nc2)=O)C2CC2)=O)sc(C)c(Br)c1C 27249,Cc1ccc(C(N2CC=CC(NC(c3cccn3C)=O)C2)=O)c(F)c1F 27250,c1(C(=O)NC2CCN(C(C3C(=C)C3)=O)CC2F)c(C)c2cc(O)ccc2oc1=O 27251,c1(N(C(c2nc(C3N(C(C(COC)O)=O)CCC3)sc2)=O)CCO)ccc(C)cc1 27252,c1(C(=O)NC2CCN(C(c3c(SC)ccs3)=O)C2)cc2c(cn1)OCCC2 27253,C1(NC(c2cn(CCC)nn2)=O)(CO)CCCN(C(C2(F)CC=CC2)=O)C1 27254,CCC(CC)C(C)C(=O)NCCCC(C)(C)NC(C1CCC(C)O1)=O 27255,N1(C(C(C)NC(C)=O)=O)CC2CN(Cc3ncnn3C(C)C)CC2C1 27256,c1(C(=O)NC2(C)CC(NC(C3(C)N(C)CC(O)C3)=O)C2)cc(F)c(Cl)cc1F 27257,N1(C(C(CSC)C)=O)CCCCCC(NC(c2cc(C)cnc2C)=O)C1 27258,c1(C(N(C(CCNC(C(C(C)O)(F)F)=O)C)C)=O)ccc2c(c1)N(C)C(=O)C2 27259,C(C(N=[N+]=[N-])C(=O)NC1CCN(S(=O)(=O)C(F)F)CC1)OCC 27260,N1C(NCC(C)(C)C#N)=NCCC(C)CCC1 27261,C1(C)(CNC(c2c(C)nco2)=O)CCN(C(=O)CSCc2cccnc2)CC1 27262,C(C(C(C)(C)C)NC(C1(O)CC1)=O)NC(c1cc(C(=O)OC)sn1)=O 27263,C1(NC(C(C)NS(CC)(=O)=O)=O)(CF)CCN(C(c2c[nH]nc2C(=O)OC)=O)C1 27264,C(=O)(CC(=O)N(CC(=O)N(C1CC1(C)C)C)C1CC1)NCC 27265,c1(CC=CCC(=O)NCCCCN(C)C(C2CCC3CC23)=O)ccccc1 27266,C(C(CC(C)C)C(=O)NC(c1ccccc1)CO)NC(c1cnn(C=C)c1N)=O 27267,CCC(CC(=O)NCC1COCCN(C(=O)C(F)C2CCC2)C1)CC(C)C 27268,CCC(C)(C)CCCC(=O)NCC1CCN(C(=O)C#CC(=O)N(C)C)CC1C 27269,Cc1ccc(C2(C(=O)NCC3CCCN3C(=O)C=CC(=O)N(C)C)CCC2)cc1 27270,Cc1cc(C)c(C(=O)NCC(C)C(=O)NCCc2nccs2)s1 27271,C1(OC)(CNC(=O)C(C)c2ccsc2)CN(C(=O)CC2CC(=O)C2)C1 27272,C1(CCNC(CSCC=C)=O)CCCN(C(=O)C(C)Cn2ccc(C)n2)C1 27273,C(=O)(C#CC(C)(C)C)Nc1ccccc1-n1cncn1.C12CCN(C1)C2C 27274,c1(C(N(C(CSC)C)C)=O)cn(C2CCCNC2)nn1 27275,C1(NC(C(=O)N(CCC#C)C)=O)CNCC12CC2 27276,Cc1ncc(C(=O)NCC2CC(F)CN2C(=O)CC2CCOC2=O)n1C(F)F 27277,c1(N2CCC(OCC)CC2)nc(=NCc2cc[nH]c(=N)c2)[nH]c2c(C)nn(C)c12 27278,CCCCC(F)(F)C(=O)NCCC1CCCN1C(=O)CC1CNC(=O)O1 27279,C(CC(C)C(=O)N1CC(c2ocnc2CNC(c2sccc2C)=O)C1)OC 27280,c1(NC(C(C)(C)c2cncs2)=O)nc(O)ccc1-c1ccccc1 27281,C1(C(=O)NC2CCC(C)(C)C2)CC12CCSCC2 27282,c1(CC)cc(CC)nc(N2CC3C(CNC(=O)C(c4cnn(C)c4)C)C3C2)n1 27283,N1(C(COCCCC)=O)CC2CCC(CNC(C3CC3(C)CC)=O)(C2)C1 27284,C(C(CO)C(C)CC)NC(C1C(CCC)CN(C(=O)C(C)(C)N(C)C)C1)=O 27285,C1(CC(=O)NCC2CCCCS2)CCN(C(c2cc(Cl)ns2)=O)CC1 27286,C12(C(N3CCC(C(C)NC(c4cccc(N)n4)=O)C3)=O)CC3CC1(CO)CC3C2 27287,C1(C(N)=O)CCN(c2nnnn2-c2nc3c(s2)CCC3)CC1O 27288,c1(C(=O)NCC(CCCC)NC(c2ccc[nH]2)=O)cnc(O)c2ccsc12 27289,C(=O)(CC(C(C)(C)C)NC(c1cc(F)ccc1F)=O)N(CCN=[N+]=[N-])C 27290,N1(C(Cc2nc(C)sc2)=O)CCN(C(c2sc(C3CC3)nc2C)=O)CC1C1CC1 27291,N1(C(C(C)(C)O)=O)CCCC(C(N2CCC(COC(F)(F)F)CC2)=O)CC1 27292,Cc1nn(-c2ccncc2)cc1C(=O)NCCC(O)CNC(=O)C(C)(C)CF 27293,C(=O)(CCC(=O)N(C(CNC(=O)CCCCN1CCCCC1)C1CC1)C)NC 27294,CCCCCC(C)CC(=O)NCc1cc(C(=O)N(c2cccc(C)c2C)C)cs1 27295,C(=O)(CC(CC)CC(C)C)NC(CCC(=O)NCCC(=O)NCC(C)C)C(C)C 27296,N1(c2ccnc(COC)n2)C2CCC1(CNC(c1cccc(F)c1F)=O)CC2 27297,c1(C(=O)NC2CC(F)(CNC(=O)C=Cc3cc[nH]n3)C2)cc2ccsc2s1 27298,c1(OC)ccc(C(N2CCN(C(c3c[nH]ccc3=O)=O)C(C)C2)=O)cc1F 27299,CCC(CCC(=O)NCC(O)Cn1cccn1)NC(c1nc(CC)oc1C)=O 27300,C1(NC(C(C)c2ccco2)=O)CN(C(=O)C=CC2(C)COC2)CC1C1CC1 27301,N1(C(C(C)(C)CF)=O)CCOCC(C)(CNC(c2ccccc2)=O)C1 27302,Cc1cnc(CNC(=O)CC2CCN(C(=O)C(c3ccccc3)C3CC3)C2)o1 27303,C12(NC(CC(CC)SC)=O)CCCCC1CN(C(=O)CCCS(N)(=O)=O)C2 27304,N1(C(C(C)n2cncn2)=O)CC2CC2(C(=O)NOCCF)C1 27305,CC(c1ccccc1)=CC(=O)NC(CC(=O)N1CCC(C)C1)C(F)F 27306,c1(N2CCC(CNC(C(C3CCOC3)OCC)=O)CC2)cccc(F)c1C#N 27307,C1(C(N2C(C(C)NC(c3c(C)csn3)=O)CCC2)=O)CCCN(C)C1 27308,c1(C(C(=O)NCC2CCN(C(=O)C=Cc3nccs3)C2)O)cc(Cl)cc(Cl)c1 27309,C1(NC(c2c(C)ncnc2)=O)(CO)CCCN(C(c2ccccc2Br)=O)C1 27310,C=CCCCCCC(=O)N1CCCC(C(C)NC(=O)C2CC2)C1 27311,Cc1sc2ncc(C(N3CC(CC(C)NC(C4(C)CCCC4C)=O)C3)=O)n2c1C 27312,C1(SC)CN(C(C2(OC(C)C)CCCCC2)=O)CC1NC(=O)C=C(C)C 27313,C(=O)(C1=NOC(C)C1C)N1CC2C(CC(N3CCC(SCC)CC3)=O)(CC2)C1 27314,N1(C(CCC(C)(F)F)=O)CCc2sc(CNC(=O)C(=C3CCCCC3)F)nc2C1 27315,C1(C(=O)NC23C(CN(C(C4(C)COC4)=O)C2)C3)CS(=O)(=O)CC12CC2 27316,c1(C(N2CCN(C(C(C(C)C)C)=O)CC2C2CCC2)=O)cccc2ccnn12 27317,N1(C(C(CC(F)F)NC(=O)C(C2CC2)C2CC2)=O)CCN2C(=O)OCC2C1 27318,C#Cc1cncc(CN2CCN(C(=O)CN3CCCCC3)C(CC)C2)c1 27319,N1(C(CCOCCOC)=O)CCC(C)C(N(C)C(c2ccc(OC)cc2C)=O)C1 27320,c1(CCC)ccc(C(=O)NCC(C(C)C)NC(=O)C(C)CSC)cc1[N+](=O)[O-] 27321,C(=O)(CC1=CCOCC1)NC(C1CC(NC(C2CCCC2(F)F)=O)C1)C 27322,CC(C)CCCC(C)CNC(C1CC(C)CN(C(c2cncc(F)c2)=O)C1)=O 27323,CCCCC(C)(F)C(=O)NCC1CCC1NC(=O)C1=CCCCO1 27324,c1(-c2c(C)n[nH]c2)ccc(C2(NC(C3CCC(=O)N3)=O)CC2)c(F)c1 27325,c1(C(=O)NCC2C(C)(C)C(NC(=O)Cc3cc(Cl)cs3)C2)cncc2[nH]ccc12 27326,C(=O)(C(F)(F)C1CC1)NCCNC(C1(n2cncn2)CC1)=O 27327,N1(C(C(COC)C)=O)CCCC(O)(CNC(c2ccc(C(F)(F)F)cc2Cl)=O)C1 27328,C(=O)(C(C)C(C)(C)O)N(C1CCCN(C(CCSc2c(OC)cccc2)=O)C1)C 27329,c1(C(=O)NCCCC2N(C(CC(C)SC)=O)CCCC2)cccc2nncn12 27330,c1(C(C)C)n[nH]cc1C(=O)NCC(O)CN(C(=O)CCc1ccsc1Cl)C 27331,C1(NC(c2csc(C)c2C2CC2)=O)CCCC12CN(C(=O)Cn1ccnc1C)C2 27332,C(=O)(CC(C)(C)C#N)N.c12ccoc1C(=O)NCC(C)(C1(C)CC1)NC2=O 27333,c1(C(CNC(=O)CCc2cnccn2)NC(CC2CC(=O)C2)=O)ccccc1 27334,C1(CNC(CCC=CC)=O)CN(C(=O)C(C)Cc2ccncc2)CC2(CCC2)O1 27335,N1(C(C(CSC)O)=O)CCCC12CCC(NC(=O)CN(C)C)CC2 27336,C1(C(N(C2CN(C(=O)CSc3ccn(C)n3)C2)C)=O)CCn2ccnc2C1 27337,N1(CC(=O)NC(C2CSC2)C)C(C)CCC1C 27338,CC(C(CO)NC(=O)CCc1cncn1C)NC(c1cn(C2CCC2)nn1)=O 27339,c1(C(N(c2ccccc2)CCCC)=O)ccc2c(c1)CNC2=O 27340,C1(NC(C(CSC)C)=O)CCSC12CN(C(=O)CCc1ccc(O)c(F)c1)C2 27341,CCCCCC(CC)C(=O)NC1CCC1CNC(=O)CCCNC(=O)C(C)(C)C 27342,c1(C(N2C(C)(C(=O)Nc3cccc(OC)c3)CCC2)=O)cc(Cl)cnc1Cl 27343,C(=O)(C(CN=[N+]=[N-])NC(=O)C(C)NC(=O)N(C)C)NC(c1cn[nH]c1)C 27344,C1(C(=O)NC2(CC)CCCN(C(CNC(CC)=O)=O)C2)CCC2(CCC2)CC1 27345,c1(OC)ccc(C(=O)NC2CC2NC(c2cc(C)cc(F)c2)=O)cc1C1CC1 27346,CC1(CNC(=O)CN2CC=CC2)CC(NC(c2ncsc2Br)=O)C1 27347,Cc1noc(C(C)C)c1C(=O)N(C)CC1(O)CCN(C(=O)CC(C)NC(N)=O)C1 27348,c1(C(=O)NC(C(C)NC(c2cc(N)cnc2Cl)=O)C)ccc(Cl)c2ccccc12 27349,C12(C(=O)OC)CCCC1CCN2CCn1cnnc1 27350,C1(C(C(=O)OC)O)CCN(C(=O)NCc2c[nH]nc2C(C)C)CC1 27351,CC1CN(C(=O)C2=COCCC2)CC(C(=O)NC2(C)CC(O)C2)O1 27352,c1(C(=O)NC2CC2NC(c2noc3c2CCCC3)=O)ccc2cccnc2c1 27353,Cc1nn(Cc2ccccc2Cl)c(Cl)c1C(=O)OCC1C(C)(C)C1(F)F 27354,c1(NC)ccc(C(N2CCC(CC)C2C(N2CC(OC(=N)O)C2)=O)=O)cc1 27355,C(=O)(CCCCC(=O)N1CC(O)(C(F)C(=O)N(C)C(C)C2CC2)C1)OC 27356,CC1(F)CCC(C(N2CCC(CNC(=O)C(F)(F)c3cncs3)C2)=O)CC1 27357,CC(C)C(CC(=O)NCC(C)CNC(c1cnc(C2CCC2)s1)=O)C(C)C 27358,CC#CCCCC(=O)N1CC(C(=O)NC(CC2CC2)C(=O)OC)C(F)(F)C1 27359,c1(CNC(C(C)O)=O)ccc2c(c1)CCN(C(c1coc(CO)c1)=O)C2 27360,C1(C)(CNC(C2(C)C(C)CCC2)=O)CCCN(C(c2ccc(F)s2)=O)C1 27361,C1(C(=O)NCC2N(C(Cc3ccc(C)o3)=O)CCC2C)CCc2nncn2C1 27362,N1(C(C=CCC(C)NC(C2(O)CCCCC2)=O)=O)CC(CO)CC12CCC2 27363,c1(OC)cccnc1C(=O)NC1(C)CC(NC(=O)CCC2CCCO2)C1 27364,c1(CC)c(C(=O)N(CC(C)NC(=O)CC2(O)CCCC2)CC)cnn1CC(C)C 27365,Cc1ccc(-c2cc(F)c(F)cc2O)c2nc(C(=O)NC3CNC(=O)C3)cn12 27366,C(C)(C)(CC=CC(=O)NC1CC(CO)C1)NC(CCOC)=O 27367,C(=O)(C1=COCCO1)N(C(CCC(=O)NCCCC(C)O)=O)C 27368,C(=O)(C(CO)NC(C1CCCN1CCC)=O)NCC=C 27369,c1(C(=O)NC2CCCC2c2nc(S)n[nH]2)cc(O)nc(C2CC2)n1 27370,C1(CC)CN(C(c2cc(C)oc2C)=O)CCC1NC(c1cnn(CC(F)F)c1)=O 27371,Cc1ncnc(C)c1C(=O)NCC12CC(CO1)N(C(=O)C=Cc1ccc[nH]1)C2 27372,c1(N(C)C(c2c(F)cccc2Cl)=O)ncnc2ccccc12.C12CCN(C1)C2 27373,c1(NC(C)=O)cccc(C(N2CC(O)(C(C)NC(C3CC34CCCC4)=O)C2)=O)n1 27374,Cc1cc(C)c(C(=O)NC(C)(C)CCCNC(C2CCCC(F)C2)=O)[nH]1 27375,CCCC(C)(C)C(=O)N1CCC(C)(NC(=O)C(N2CCC(C)C2C(=O)OC)=O)C1 27376,C1(C(=O)NCc2ccc(F)nc2F)CC12CCN(C(c1cc(O)ccn1)=O)C2 27377,C#Cc1cccc(CNC(=O)C=C(C)CNC(=O)C(C)(C)C(N)=O)c1 27378,C#Cc1cn(C)nc1C(N1CCC(C(N2CC(O)CC2(C)CO)=O)C1)=O 27379,C(=O)(CCC(=O)c1ccncc1)N(C1CCN(C(=O)C(=O)NCC2CC2)C1)CC 27380,C1(C(=O)NCCNC(c2c(OCC)oc(C)n2)=O)CC1C1CC(F)(F)C1 27381,c1(SCCC(=O)NC2CC(C)(NC(C(CCN(C)C)O)=O)C2)cc(F)ccc1F 27382,C(CC#C)(CC(=O)NC1(n2cc(-c3ccc(F)cc3)nn2)CCOCC1)NC 27383,C(=O)(CC(O)CC(C)C)NC(C(=O)NC(C#C)C)C1(C)CC1 27384,Cc1ccccc1OCCC(=O)NCCCc1nccs1 27385,Cc1cc(C)c(C(N2CC(O)(CCNC(C3(C4CCC4)CC3)=O)C2)=O)s1 27386,c1(OC)ncccc1-c1cnc(CC(=O)NCC2(C(F)(F)F)CCC2)nc1 27387,c1(C(=O)NCC#CCC(=O)NCCC(COC)O)ccc2c(c1)CCC2 27388,C1(C(N2CC(C(=O)NC(C#C)CC3CC3)(CC=C)C2)=O)CCCC(O)C1 27389,c1(C(N(C2C(N(C(C=C(COC)C)=O)C)CCCC2)C)=O)cnc2sccn12 27390,N1(CC(N)=O)CCN(C(=O)C(=O)NCCCN2CCCCCC2)CC1 27391,CC(C)C(C(=O)Nc1cncc(C#N)c1)C(C)NC(C1CC(O)C1)=O 27392,C1(C(=O)NC2CC3CC(NC(C4=CC(C)(C)C4)=O)CC32)COc2ccccc2O1 27393,C(=O)(C(C)CC(N)=O)NCc1cn(CC2N(C(CSCCOC)=O)CC=C2)nn1 27394,C(=O)(C(C)CN(C(=O)CC1CNC(=O)O1)C)NC1CC(CSC)C1 27395,N1(C(C2CC(C)C2)=O)CCOC(C(=O)NC2CCC3(C(=O)OC)CC23)CC1 27396,C1(CC(N2CCC(CC=C)C2)=O)CN(C(c2cc(O)n(C)n2)=O)CC1C 27397,Cc1c(C(=O)NCC(C(C)C)NC(=O)COC(F)F)cnn1CCC(C)C 27398,CC(C)CCC(F)C(=O)N1CCC2(CC2C(N2CC3(CCOC3=O)C2)=O)C1 27399,c1(C(N(CC(C)(C)CNC(C2(CC)CCCC2)=O)CC)=O)cc(C)cc(O)c1 27400,c1(CC(=O)NCCCC(C)NC(=O)CC2CCN(C)C2)ccc(N)cn1 27401,N1(C(c2c(OC)csc2)=O)CC(OC)CC1C(=O)NCCN1CCC2CC12 27402,C=CC(C)C(C)C(=O)NCCCN(C)C(c1cncc(C#N)c1)=O 27403,C1(C)(CNC(Cn2c(C)nnn2)=O)COCCN(C(c2c[nH]cc(Cl)c2=O)=O)C1 27404,CC1(NC(=O)Cn2cnnn2)CC(NC(C2(c3cccs3)CC2)=O)C1 27405,Cc1cccc2nc(NC(C3CCN(c4cccc(Br)n4)C3)=O)[nH]c12 27406,c1(CC(=O)NCCC2CCCCN2C(=O)C=C2CCC2)n[nH]c2ccccc12 27407,c1(OC)ccc2ccccc2c1CNC12CC(NC(c3c[nH]nc3C)=O)(C1)C2 27408,C1(C)(CNC(c2cn(C)nc2)=O)CC(F)(F)CN1C(c1cnc(C(C)(C)C)[nH]1)=O 27409,c1(OCC)ncccc1CN1CC2CC2(C(=O)NCc2ccccc2Br)C1 27410,C1(N(C)C(C2(C3CC3)CCCO2)=O)CCN(C(c2ccc(CO)nc2)=O)CC1 27411,S(=O)(=O)(c1cc(F)ccc1F)N1C(C(=O)Nc2ccc(Br)nc2F)C2CCC1C2 27412,N1(C(CCC=C)=O)CCC(C(N2CCC(N3CCC3)CC2)=O)C(C)(C)C1 27413,C(C)(C)(CCC(=O)Nc1ccccc1O)NC(CCC1N(C)CCC1)=O 27414,N#Cc1ccc(S(N)(=O)=O)c(N2CC3CC2C2OCCOC32)c1 27415,C1(O)(CNC(C2(C(=O)OCC)CC2)=O)CCN(C(=O)C(N2CCC(O)CC2)C)C1 27416,n1(C(C)C)cnc(C(=O)NCC(C)(C)NC(=O)C(C)NC(c2cccs2)=O)n1 27417,C(C1CCCCCC1)=CC(N1C(CNC(c2c(C)noc2C(F)F)=O)CCC1)=O 27418,C1(O)(CNC(CCCN(C)C)=O)CCCN(C(=O)CC2CCC(C)(C)CO2)C1 27419,Cn1cc2c(C(=O)NCc3cccc(Br)c3Cl)cc(C(F)(F)F)cc2n1 27420,N1(C(C2(CCC=C)CN(C(=O)C=CC(=O)N(C)C)C2)=O)CCS(=O)C(C)C1 27421,CC1CN(C(=O)CC2C3CCCC3N2C(=O)COCCCF)C2(CC2)C(=O)N1 27422,c1(CC)cccc(OCC(=O)N(CCCNC(C2CCC(C)O2)=O)CC)c1 27423,CC1(C)COC(C(=O)NC2CCC(CC(N3CCOCC3CO)=O)C2)C1 27424,C1(NC(C(C)CC2CCCCC2)=O)CCN(CCCN(C)C)CC1C 27425,c1(C(=O)NCCCN(C(c2ccc(Br)cc2F)=O)CC)ccc2c(n1)CCO2 27426,C(CC(C)C(=O)NCc1ncoc1CCNC(C1CC1F)=O)=CCC 27427,CC(C)C(CCN(C)C(c1occc1CN(C)C)=O)NC(C1(C)CCSCC1)=O 27428,N1(C(C2CC(SC)C2)=O)CCN(C(c2ccnn2C2CCOCC2)=O)CC1 27429,N1(C(C2CCC(=O)OCC2)=O)CC2(CCCN(C(C3CN4CCC3CC4)=O)C2)C1 27430,N1(C(COC2(C)CCC2)=O)CCOC(C(C)NC(c2ccc(C(N)=O)[nH]2)=O)C1 27431,C1(C)(C(=O)NCc2cn(C(CC)C)nn2)CCC2CC2C1 27432,C1(NC(c2cc(COC)no2)=O)CCN(C(=O)C(F)(F)C(F)(F)F)CC12CCC2 27433,c1(CC(=O)NC2CC(F)(CNC(c3cn[nH]c3)=O)C2)cccc2ccccc12 27434,Cn1nc(C(=O)NCc2cc(Br)co2)c2c1CNCC2 27435,C(=O)(C1CCCn2cnnc21)N(CCCNC(C1CC2(C1)CC21CCC1)=O)CC 27436,C(=O)(C(O)C(C)(C)CC)NCCCOCCC(NOCCC(=C)C)=O 27437,C1CCCC(=O)N(c2nc[nH]n2)Cc2ccc(s2)N1.C1(OC)(CO)CC1 27438,CC(C(=O)NC1COCCN(C(C2CN3CCCC2C3)=O)C1)S(C)(=O)=O 27439,C(CC(=O)NC(c1ccccc1C)C)(C(F)(F)F)NC(CC(C=C)C)=O 27440,CC1(C(=O)NCC2CCCC(NC(=O)COCCc3cccs3)C2)CNC(=O)C1 27441,C1(CC=C)(C(=O)NCC(CO)NC(C2CCCN2CC)=O)CCCCC1 27442,c1(C(N2C(CNC(CC(CC)C3CC3)=O)CCC2)=O)ccc(OC)c2ccsc12 27443,c1(CNC(C2CC(N(C(C(C)=CC=C)=O)C)C2)=O)ccc(C)s1 27444,C1(CNC(Cc2c(C)non2)=O)CCCN(C(C2SCCS2)=O)CC1 27445,N1(C(Cc2n[nH]c(=N)s2)=O)CC2CC1CCC2NC(c1cncc(C2CC2)c1)=O 27446,c1(OC)ccc(O)cc1C(=O)NCC(C)CNC(=O)CC(C)=C(C)C 27447,c1(NCC(C2CCCC2)NC(c2ccn(C)n2)=O)ncc2c(ncn2C)n1 27448,c1(N2CCN(C)C(CNC(c3cccc(C(F)F)n3)=O)C2)ncc(C#N)cc1F 27449,c1(CC)ccsc1C(=O)NCC=CC(=O)N(C1CCSC1)CC 27450,c1(CN(CCCO)C(=O)Nc2cc(-n3cccc3)ccn2)ccc(Cl)cc1 27451,c1(C(N2CC(CC(=O)Nc3cnc(Cl)nc3)OCC2)=O)cnn2ccccc12 27452,C1(CC(=O)OC(C)(C)C)COCCN1C(=O)C=O.N1(CCOC)CCN(CCO)CC1 27453,C(=O)(C#CC1CCCC1)N1CCN(C)C(C(N2CCC(F)(CF)C2)=O)C1 27454,C1(NC(N2C(C)CSCC2)=O)CCCN(S(=O)(=O)N2CCOCC2)C1 27455,N1(C(c2ccc(SC)s2)=O)CC2CCCC2(CNC(=O)CCCC#N)C1 27456,Cc1[nH]nc(Br)c1C(=O)NC(C1CCCN1C(=O)CCc1cc[nH]n1)(C)C 27457,c1(OC)ccc(CCC(=O)NC2CC(C)(NC(C3CCCC3(C)C)=O)C2)cc1F 27458,C1(NC(C(CC)SC)=O)CC1C1CCCN(C(=O)C(=O)C(F)(F)F)C1 27459,C(=O)(C(CO)C(F)(F)F)N1C(CCC(=O)NCCOCC#C)CCC1 27460,N1(C(CNC(CNC(c2ccc(C)cc2)=O)=O)=O)CCC2C(C(N)=O)C2C1 27461,Cc1cc(C(N2CCC(NC(c3cc(F)c(Cl)cc3Cl)=O)C2C)=O)cc(F)c1C 27462,c1(C(=O)NCCCN(C(c2nc(Cl)cs2)=O)CC)ccnc(C(C)(F)F)c1 27463,CC1(CF)CN(C(C2(C3CCCN3C(c3cncs3)=O)CC2)=O)C1 27464,C(CCC(O)C(=O)NC(C)C(=O)NCC(C)C)NC(C(C=C)CC)=O 27465,N1(C(CC(COC)C)=O)CC2CCN(C(c3cnn4c3OCC4)=O)CCC2C1 27466,CC1OC2(CNC(C3C(C)OC(C)C3C)=O)CC1(NC(C1CCCOCC1)=O)C2 27467,CCCCCCC(C)NC(=O)C1=CCN(C(=O)CCC2CCCO2)C1 27468,S(=O)(=O)(c1ccc(NCCCCS(C)=O)nc1)N(C)Cc1scc(C)c1 27469,Cc1ccc(C(N2CCCCC(CNC(c3n[nH]c(C4CC4)n3)=O)C2)=O)nc1O 27470,C(c1csc(C)n1)=CC(=O)NC(CC=C)CNC(c1cc(CF)on1)=O 27471,C1(C(=O)NCC2C(C)C2C)CCN(C(c2ncccc2Cl)=O)C1(C)C 27472,c1(C(N2CCOCC(C(N(CCC(=O)NC)C(C)C)=O)C2)=O)cccc2ccoc12 27473,C1(CC(=O)N(CC(O)CNC(=O)C=Cc2cccs2)C)CCC(F)(F)CC1 27474,c1(NC(C(=O)NC(c2c(C)cccc2C)C)=O)ccc2c(c1)CCC2 27475,c1(C(N2CCC(N(C(=O)CC3C=CCC3)CC#C)C2)=O)ncc(OC)nc1OC 27476,C1(NC(CNC(N)=O)=O)(CNC(c2ccn(C3CCCCC3)n2)=O)CCOC1 27477,CCCCC(CC)C(=O)NC1(CC(=O)NC2CCOC2C2CC2)CCC1 27478,c1(CN2CC(C)(CC(=O)Nc3ccnc(C(N)=O)c3)C2)ccc(Br)cc1[N+](=O)[O-] 27479,CC1(C)OCCC1C(=O)NCCn1ccc(C(N2CCC3CC23)=O)c1 27480,C1(NC(C=CC)=O)CC=C(C(=O)NCc2cnc(CC)[nH]2)C1 27481,C(=O)(CC(C)(C)C(=O)N(CCCNC(=O)C(C)CSC)C(C)C)OC 27482,c1(C(N(C(c2cccc(Cl)c2)C(=O)OC)C)=O)cc(Br)cc(I)c1C 27483,C(CCCC)(CN=c1[nH]c(Cl)ncc1C(C)C)NC(C=CC(=O)NCCCC)=O 27484,c1(CCC(c2n(CCOCC)nnn2)NC2CC(C)(C)C2)cccc(Br)c1 27485,C1(NC(CN(C)CC)=O)CC(NC(c2cc(C(C)C)ccc2C)=O)C12CCC2 27486,c1(C(N2CC(NC(=O)CN(C)C)CC(OC)C2)=O)ccc2c(=O)ccoc2c1 27487,C(=O)(C(C)CC(C)C)N1CCC(C)(CC(=O)NCCNC(=O)OCC)C1 27488,Cc1c(NC(c2oc(CNC(=O)CC3CCC(C)C3)nc2C)=O)cnn1C(C)C 27489,c1(C(C(F)F)NC(=O)Nc2cn(C(C)(C)C)nc2)ccc(F)cc1F 27490,C(=O)(CN=c1cc[nH]cc1)NCCCCCNC(=O)CCC(=O)c1cccnc1 27491,C1(C(N(CC(=O)OC)C)=O)(C(C)C)CCCN1C(c1ncn(C(C)C)n1)=O 27492,N1(C(c2cc(=O)c(Cn3cc(CCCO)nn3)co2)=O)CCn2cncc2C1 27493,c1(N2CC(O)(C(C)NC(=O)CCc3ccncn3)C2)nc2c(F)cccc2o1 27494,C1(NC(CCc2cnn(C)n2)=O)CN(C(=O)C=C(Cl)Cl)CC1N=[N+]=[N-] 27495,Cc1cc(Cl)c(CN2CCCC2CC(N2CCC(C)(O)CC2)=O)c(Cl)c1 27496,C(C(C)(CCO)NC(C1CCCCN1C(c1snc(C)c1N)=O)=O)OC 27497,c1(OCCC(=O)N(CCN=[N+]=[N-])CCOC)ccc(C)cc1Br 27498,C1(CNC(C(c2cn(C)nc2)=O)=O)CCCCCN1C(c1ccsc1Cl)=O 27499,c1(CNC(C=CCC2(NC(c3n(C)ncn3)=O)CCC2)=O)cc(=O)cc[nH]1 27500,CC1(C)CN(C(C2(CCNC(c3ccc(=N)[nH]n3)=O)CC2)=O)CCC1O 27501,c1(C(N2CC3C(NC(C4C(CCC)C4)=O)(CC3)C2)=O)cc(S(C)(=O)=O)co1 27502,N1(CC(CCC)(C)C)CCC(O)C(C(=O)N(C)Cc2cccc(OC)n2)C1 27503,CCC(C)(CC)C(=O)NCCNC(C1CN(C(C23CCC(C2)OC3C)=O)C1)=O 27504,c1(C(N(C2CCN(C(C34C(=O)C5CC3C4C5)=O)C2)CC)=O)cc(=O)n(C)cn1 27505,CC(C)C(CNC(=O)COCc1ccccc1)NC(=O)CCc1cc(Cl)no1 27506,c1(OC)cc(C(N2CCC(CNC(c3ccc(CF)cc3)=O)C2)=O)cc(F)n1 27507,C(=O)(C1=C(Cl)CCCC1)N(C(C(=O)NCC(C)N(C)C)CO)C 27508,CCCC(CC)CCC(=O)NC1C=CC(C(N2CCC(O)C2C)=O)C1 27509,C1(C(=O)NCC2(O)CC(CF)C2)(COC)C=CCN1C(=O)CC1COCCOC1 27510,CCC(CC(=O)NC1CCC(NC(c2cc(F)cc(Cl)c2)=O)CC1)C(F)F 27511,N(C1COc2ccccc21)C(CC1CCN(C(c2cc(C)ns2)=O)C1)=O 27512,CCCC(C(=O)NC(C(=O)NOCCN1CCCC1=O)C1(O)CCC1)C(C)C 27513,Nc1c(C(=O)NC2CC(NC(C3(F)CCC3)=O)C2)cc(Cl)cc1F 27514,c1(CC(C)(CO)N(CC(O)C2CCC2)C)cccc(Br)c1 27515,C#Cc1cc(C(=O)NCCC(C)NC(c2csc(C#N)c2)=O)cc(C(F)(F)F)c1 27516,C12(C(=O)OC)CCC(C(CC3=CCS(=O)(=O)C3)=O)(C1)OC2 27517,N1(C(c2cc(COC)cn2C)=O)CCN(C(=O)CN2CCSCC2)CC1CF 27518,c1(NCC(C)F)[nH]c(=NC(CC2CC2)c2ccccc2Cl)nc2sccc12 27519,C1(N(C(c2c(OC)csc2)=O)C)CCCC2CN(C(C3CCN(C)C3=O)=O)CC12 27520,C1(CC=C)(NC(COCC=C)=O)CN(C(=O)Cc2cc(-c3ccccc3)on2)C1 27521,c1(C(=O)NCC(CNC(=O)CC2(O)CCOC2)O)ccc2ccccc2n1 27522,C1(CNC(CC(C)OC)=O)CC2(CCC2)CN1C(C1CN(CC(F)(F)F)C1)=O 27523,C1(C(=O)NCC2CCCC(CNC(C3(C)CS(=O)(=O)C3)=O)C2)C(F)(F)C12CCC2 27524,c1(NCCCCC(C)NC(=O)CC2CCCCC2O)c([N+](=O)[O-])cnn1C 27525,CC1CCC(C)(C(=O)NCCCOCCNC(=O)CCc2cc(Cl)no2)C1 27526,C1(C(=O)NC2COCCN(C(=O)Cc3ccoc3)C2)CC2(C1)CC(F)(F)C2 27527,CC1(C)CN(C(C2CCCOC2)=O)CC(C)(C)C1NC(C1CC(C(F)F)C1)=O 27528,c1(C(=O)NC)ccc(C(=O)NC2CN(C(C3COCCO3)=O)CCC2F)cc1F 27529,C1(C(N2CCC(OCC)C2)=O)CC2(CC2)CN1C(=O)CC1CCC=CCC1 27530,C1(NC(C=CSC)=O)CCCCC12CCCN(c1cccc(SC)c1[N+](=O)[O-])C2 27531,CCC(CO)CN=c1[nH]c(=NCc2cc(F)c(F)c(F)c2)c2sccc2[nH]1 27532,C#CC(C)(C)C(=O)NCCCC1CN(C(c2ccc(CC(N)=O)cc2)=O)CCO1 27533,c1(C(N2CC(C(=O)N(C3CC3)CC3CC3)OCC2)=O)cccc2[nH]ccc12 27534,c1(OC)cc(NC(C2(CNC(C3(C)C=CCCC3)=O)CC(OC)C2)=O)cc(F)c1 27535,c1(C(N(CCC(C)NC(=O)C=Cc2nccs2)C)=O)cc(-c2cccs2)[nH]n1 27536,c1(C(N2CC(O)(C(C)NC(CC(C)C(F)F)=O)C2)=O)cnc2c(c1)NC(=O)CO2 27537,c1(CCNC(N(C2CC(OCCCCC)C2)C)=O)c[nH]c2cc(F)ccc12 27538,Cc1cc(C(=O)NC2CCC(C(=O)NCC3(CC4CC4)CCC3)C2)c(C)o1 27539,Cc1nc2c(o1)CCCC2CC(=O)N1CC2CCC1CN2C(=O)Cn1cncn1 27540,C1(C(N(C)CC2(C)CCCO2)=O)CCCCCCN1C(C12CC(C1)C2)=O 27541,C(=O)(CCCC(F)(F)F)N(CC(CC)NC(C1(C)CCC(O)CC1)=O)C 27542,CC(CC(=O)NCCC1CN(C(=O)CNC(C2CCC2)=O)C1)C(F)(F)F 27543,C1(CNC(c2cc(C)nc(O)n2)=O)CCCC2(CN(C(=O)C(C)C(C)C)C2)O1 27544,C1(CC)CN(C(=O)CC2CCCCCCC2)CCN1C(C1CC=CCO1)=O 27545,c1(C(=O)OC)cnc(Cl)cc1CN1CCC1C(=O)NCc1cccc(C)c1 27546,CC1CC(C(=O)NC2(CF)CCN(C(C3CCN(C4CCSC4)CC3)=O)C2)=NO1 27547,C1(C(=O)NC(C)C(=O)N(CC(C)(C)NC(=O)CC23CCCC2C3)C)CCCCC1 27548,c1(C(N2CCC(NC(c3cccc(OC)c3)=O)(CO)C2)=O)scc2c1OCCO2 27549,C1(NC(Cn2c(C)ccc2C)=O)CC(C(N2CC(C)(C(F)(F)F)C2)=O)C12CCC2 27550,N1(C(C(CSC)OC)=O)CCN(C(=O)C(C(C)(C)C)c2cccc(C)c2)CC1C 27551,N1(C(C2(CCOC)CCC2)=O)CC(NC(c2ccc(Cl)nc2N)=O)C2(CC2)C1 27552,N1(C(=O)NCCN(C)C(=O)NC2(c3ccco3)CC2)CCn2cnnc2C1 27553,C12(CNC(CC(=C)C)=O)CCC(CC1)N(C(c1ncc([N+](=O)[O-])n1C)=O)C2 27554,N1(C(C(C2CCN(C(c3c(CC)c[nH]c3)=O)C2)F)=O)CC=CC1(C)C(=O)OC 27555,C(=O)(CCCCN=[N+]=[N-])N1CCCC(N(C(c2c(CC)nn[nH]2)=O)CC2CC2)C1 27556,C(=O)(C(O)CC(=O)OC(C)(C)C)NC1(C)CN(C(C(CCC)C)=O)C1 27557,N1(C(C2C(C)CC=CC2)=O)CCCCC(CNC(c2cccc(F)c2N)=O)C1 27558,Cc1ccccc1C1(C)CC1NC(=O)NCCN1CC(CC#N)C1 27559,Cc1nc(C(=O)NCC(C)(O)CNC(=O)Cc2nc(=N)[nH][nH]2)c(C)n1C1CC1 27560,CC(CC(=O)NC1CC(F)(CNC(=O)CC2CC2)C1)P(C)(C)=O 27561,N1(C(COC(C)C)=O)CC(NC(C2(C)CC3CC3C2)=O)CC(O)C1 27562,N1(C(C(C(C=C)O)(C)C)=O)CCC2(CCC(CC(N3CCC(O)C3)=O)CC2)CC1 27563,C(C(C(=O)OC)NC(=O)CC(C)NC(=O)CCN1CCOC1=O)OC 27564,C(CCCCC(=O)NCC(c1ccc(F)cc1)NC(c1cccn1CC)=O)=CC 27565,CC(C)CC(C(=O)NC1(C(O)CO)CC1)NC(c1nnc(O)nc1O)=O 27566,Cc1nn2cccnc2c1C(=O)NCC12CC1CN(C(C1CCS(=O)CC1)=O)C2 27567,c1(C(C)C)c(NC(=O)NCC2CC2C(=O)OC(C)(C)C)cccc1Br 27568,C(=O)(CCCCC(C)CC)NCC(CCC)NC(c1c2c(nn1C)CCC2)=O 27569,C1(NC(c2cc(C)oc2)=O)CCC(C)(C)CC1CNC(=O)CSc1ccncc1 27570,Cc1cc(O)cc(=O)n1CC(=O)NCC1(F)CC(NC(=O)C(CN(C)C)N(C)C)C1 27571,c1(C(N2CCC(NC(C(C(CC)O)(F)F)=O)C(O)C2)=O)cc(S(N)(=O)=O)oc1C 27572,C1(C(=O)NC2C=CC(C(=O)NCCSCC)C2)COCCN1CC 27573,Cc1cnc(Cl)cc1NC(C1CCCN(C(c2cccnc2C)=O)C1)=O 27574,c1(OC)ccc(F)c(C(N2CCC2CNC(C2(O)CCCC2)=O)=O)c1F 27575,N1(C(C2C(C#C)C2)=O)CCN(C(=O)CSCc2ccccn2)CC(C)(C)C1 27576,c1(OC(C)(C)C(=O)NC2CC(C)(NC(=O)C3=NOCC3)C2)cccc(N)c1 27577,c1(C(N2CCCCC(NC(c3c(C)c[nH]n3)=O)C2)=O)cccc2nc[nH]c12 27578,c1(C(N(C)CC2CCCN(C(C(C3CCC3)OCC)=O)C2)=O)ncnc(O)c1F 27579,N1(C(C2N(C(C)=O)CSC2)=O)CCCCC(CNC(c2nc(C)nn2C)=O)CC1 27580,c1(NCC2(CO)CCCCC2)nc(N2CCCC(F)C2)nc2ccsc12 27581,c1(-n2c(C3CCCC(F)C3)nc(COCC)n2)cccc2ncccc12 27582,C(=O)(CN=c1cc[nH]cc1)N(C)CCN(C(=O)CC1CCCCO1)C 27583,c1(OC)ccc(C(=O)N(CC(C)N(C(=O)Cc2ccoc2C)C)C)nc1 27584,C1(C(=O)NCC(C)S(N)(=O)=O)C(C)OCCN1C(=O)CC1CCOC1(C)C 27585,Cc1nc(NCC2CN(C(C3C=CCC3)=O)CCC2C)ncc1[N+](=O)[O-] 27586,N1(C(COCCCOC)=O)CCCC(NC(c2cc(CO)on2)=O)C1C 27587,C(=O)(C(F)C(C)CNC(C1C=C(C)CS1)=O)NC(C(=O)OC)C 27588,CC1CN(C(c2ccc(-c3ccncc3)s2)=O)CC(C)C1NC(c1cc[nH]c1)=O 27589,C1(CC)NC(=O)N(CC(=O)Nc2cc(C3CCCCC3)no2)C1=O 27590,Cn1c(CNC2(c3noc(C(F)(F)F)n3)CCCC2)cc2sccc12 27591,c1(C(=O)NCC2(F)CCCC2)c(-c2csc(-c3ccccc3)n2)cncc1F 27592,C(CC(C)N=c1[nH]c2cc(Cl)ccc2s1)NC(CCOc1ccc(C)cc1C)=O 27593,C1(NC(C2CN(C)C2)=O)CC(CNC(c2conc2C(F)(F)F)=O)C1(C)C 27594,N1(C(CCCC(CC)NC(CC(C(=C)C)OCC)=O)=O)CCC2CCN(C)CC12 27595,c1(C(C)C)nc2ccc(NS(=O)(=O)c3cc(Cl)sc3Cl)cc2s1 27596,C1(C(=O)Nc2c(C)n(C)nc2)CC(F)CN(C(C2CCCCN2C)=O)C1 27597,c1(C(N(C)CC2(O)CN(C(c3c(C)nc[nH]3)=O)C2)=O)[nH]c(C)c(S(N)(=O)=O)c1C 27598,C1(NC(C(C)CO)=O)CC2CCC(C1)N2C(=O)CC1=NNC(=O)C1 27599,C12(C(=O)NCC#CC)CCN(C(=O)CCc3cccs3)CCC1C2 27600,Cc1c(Br)ccc(F)c1CNC(C(=O)OC(C)(C)C)C(C)O 27601,c1(C(N2CCC(C)(O)C2)=O)cc(-c2ccco2)cc2[nH]ncc12 27602,C1(C(=O)NCC(CN(C)C(C2(F)CCCCC2)=O)(C)C)CC2C=CC1C2 27603,N1(C(C2(C)C(C)(C)C2)=O)CC2CCCC(NC(=O)CSCc3cccs3)C2C1 27604,c1(CNC(=O)Cc2ncc(Cl)s2)nc(CNC(=O)C(F)CC2CCC2)cc(O)n1 27605,C(=O)(C(C(C)CC1CCCC1)N1CCC(F)(C(=O)OC)C1)NCC(=C)C 27606,n1(CC)ccc(C(=O)NCC2CN(C(c3ncc(F)cc3N)=O)CC2C)cc1=O 27607,c1(C(N2C(CNC(c3cc(O)cc(F)c3)=O)CC2)=O)ccc(=O)n2c1CCC2 27608,CC(C)C(CCN(C)C(C1CCCC(=O)N1)=O)NC(=O)C(C1CCCCCC1)C 27609,c1(OC(C)CN(C)C(C2(C)CC=CC2)=O)cccc(N)c1 27610,CC(F)(CNC(=O)NC1CCC1C(F)F)C(F)(F)F 27611,C1(C(=O)NCC2N(C(c3cc(C)ncc3)=O)CC2)CCC2CC(C)CN2C1 27612,N1(C(CN2CCC(C)CC2)=O)CCCC(O)(CNC(=O)C(c2cncnc2)C)C1 27613,S(=O)(=O)(c1ccc([N+](=O)[O-])cc1OC)N1CC(C(=O)NC(CC)C)C(O)CC1 27614,N1(C(C(C)NC(=O)N(C)CCS(C)(=O)=O)=O)CCc2ccsc2C1 27615,N1(C(C=CC(=O)OCC)=O)CCC2(COC(CNC(c3ncccc3F)=O)C2)C1 27616,c1(C(=O)NC(C2(O)CCCCC2)C(=O)NCCSC2CCCO2)c[nH]ccc1=O 27617,N1(C(COCC(=O)OC)=O)C(C(=O)NCc2conc2C(C)C)CC2CCCC12 27618,c1(CCC#N)ccc(C(=O)OCc2cccs2)cc1 27619,C12(C(=O)OC)CC(NCc3ccccc3)C1C2.C1CO1 27620,N1(C(CC=Nc2c(CC=C)cccc2)=O)CCN(C(=O)CCOCC)CC12CC2 27621,c1(C(=O)NCc2c(C#N)cc(F)cc2)n[nH]c2cc(C3=CCCCC3)ccc12 27622,C(C(=O)NCc1ocnc1C(=O)NCC1(F)CC(O)C1)(C(C)C)SC 27623,Cc1cccc(C(=O)NC2CCC(NC(C3CSCN3C(=O)C(C)C)=O)C2)c1F 27624,Cc1nocc1C(=O)NCC(C1CCCC1)NC(=O)C(C)c1ccco1 27625,N1(C(CCSc2n(C)cnn2)=O)CCCC(CNC(=O)COC2CCOC2)C1 27626,N1(C(Cc2cc(CC)nn2C)=O)C2CCC1C(NC(=O)C(C)OCC(C)C)C2 27627,S(=O)(=O)(c1ccc(CCC(=O)O)cc1)N1CCC(C)CC1C(N)=O 27628,CCCCC(F)C(=O)N1CCCCC(C(=O)NCCc2ccc(C)c(C)c2)C1 27629,N1(C(C(=O)NCCC2CCCCC2(F)F)=O)CCc2ccc(Cl)c(F)c2C1 27630,N1(C(C=CC)=O)CC2CCCC2C1C(=O)N(CCC(C)C)C 27631,C1(NC(C(n2ncc(C)c2)C)=O)CCC(C)(NC(c2ccc(Cl)nc2N)=O)CC1 27632,C=CCCC(F)(F)C(=O)NC(CC)CCCC(=O)NCc1nccn1C 27633,c1(C(N2C(C)(CNC(c3cc(OCC)n[nH]3)=O)CCC2)=O)c(C)nn(C)c1F 27634,CC1CCC(CC(=O)Nc2nn(C)cc2Br)CC1C 27635,N1(C(CNC(=O)OC)=O)CC(CNC(=O)CC(C)C(F)F)C(F)(CO)C1 27636,C(=O)(C(O)CC(C)C)NCC1C(NC(C(c2ccc(CCCC)cc2)C)=O)C1 27637,C1(CNC(c2ccc(SCC)nc2)=O)CC12CCN(C(C1CCOCC1)=O)CC2 27638,CCC(C)C(O)C(C)C(=O)NC1(C(=O)NOCCc2ccccc2)CCC1 27639,C(C)(C(C(=O)N(C)CC1CCCC1)C(C)C)NC(c1snc(C)c1N)=O 27640,Cn1nccc1C(N1CC(c2ocnc2CNC(c2cnoc2)=O)C1)=O 27641,C1(CC)CC(C(=O)NCC(C)N(C(=O)C(F)OC)C)CC(=O)N1 27642,NS(=O)(=O)c1csc(C(N2CCC3C(NC(=O)CCCn4cncn4)CC23)=O)c1 27643,c1(CC)cc(C)c(C(=O)NC(C)(CNC(=O)CC2CCCOCC2)C2CCC2)o1 27644,c1(C(=O)NCCOCCNC(C(C2CCC2)OCC)=O)cc(CCO)on1 27645,N1(C(C(CCC)OC)=O)CCN(C(c2cnc(O)o2)=O)CC(CO)C1 27646,c1(C(=O)NCCOCCN(C)C(C2CCN(S(C)(=O)=O)C2)=O)cc(C(F)(F)F)c[nH]1 27647,c1(CC(N2CCC(NC(COC(CC)C)=O)C2)=O)ccc(F)cc1 27648,c1(OC)ccc(NC(C2(C)CCCN(Cc3cc(Br)co3)C2)=O)c(F)c1 27649,C1(CC)CCN(C(C)=O)C1C(=O)N(CCNC(c1scnc1C)=O)CC 27650,N1(C(c2c(SCC)cccn2)=O)CCN(C(=O)Cc2ncccc2C)CC12CC2 27651,c1(NC(c2ccoc2)C)ccc(S(=O)(=O)N(C)Cc2ccc(C#N)cc2)cc1Cl 27652,c1(C(N(CCCNC(C(C)OCC)=O)CCO)=O)cccc(CS(C)=O)c1 27653,c1(C(=O)NCCC2N(C(C3CC=C(C)CC3)=O)CCOC2)cc(C)c(C)cc1C 27654,CCCC(C(=O)N1CCOCC1CN(C)C(C1CS(=O)(=O)C1)=O)OC 27655,CC1CC(C(=O)NC2(CNC(C3(C)CC(O)CN3C)=O)CC2)=NO1 27656,N1(C(CCOCC)=O)CC(C)CN(C(c2cccc([N+](=O)[O-])c2)=O)C(C)C1 27657,c1(C(=O)NC2CN(C(Cc3cccc(C)c3)=O)CC2C(F)F)[nH]c(C)c(C)c1C 27658,C(=O)(C1=CCCCO1)C(=O)Cn1ccc(C(F)(F)F)n1.C(CN)(N(C)C=O)C1CC1 27659,Cc1cccc(CNC(=O)CC2CCN2C(=O)CN(C)C2CC2)c1F 27660,CC1CCN(C(c2cncc(O)c2)=O)CC1CNC(=O)CSc1nccn1C 27661,C(C(C(=O)N(C(C)C(C)(C)C)C)C(C)(C)C)NC(c1n(C=C)ncc1)=O 27662,C(=O)(C1=COCCC1)NCc1scc(CNC(c2c(CCC)onc2C)=O)n1 27663,CC1CN(C(c2nnn(C)c2N)=O)CCN1C(c1cccc(OC(F)F)n1)=O 27664,C(=O)(C1CCc2c(Cl)cccc21)NCC(CCCC)NC(=O)CS(=O)(=O)C1CC1 27665,C#Cc1cc(C(=O)NCC2(O)CC(NC(=O)CC3CCC3(C)C)C2)ccc1C 27666,N1(C(CCc2cnc(C)o2)=O)CC2CC1(c1cn(Cc3ccno3)nn1)C2 27667,N1(C(c2nc(C(C)(C)C)oc2)=O)CC2(CCN2C(C2C(C#N)C2(C)C)=O)C1 27668,c1(C(=O)NC2C(NC(C#CC(C)C)=O)CC2)ccc2[nH]c3c(c2c1)CCCC3 27669,C(=O)(C(F)CCC(C)C)NC1C(C)=CCS1.C12CC3(COC1C3)C(=O)N2 27670,c1(C(C(=O)NCCOC)N(C2CC3(CCC3)C2)C)nc(C)c(C)s1 27671,N1(C(C(CCC)C#N)=O)CCCC(C)(C)C1C(=O)NCC1CC(SC)C1 27672,C1(C(=O)NCCOC2CCNCC2)CC(=O)N(C2CCCCCC2)C1 27673,N#CCCCC(=O)N1CCCC1C1CCN(C(C2(C(=O)NC3CC3)CCC2)=O)CC1 27674,Cc1cc(C)n(CCNC(C2CN(C(C)C(=O)NCC3CCCO3)CCO2)=O)n1 27675,c1(C(N(CCNC(C2(CCCC)CCC2)=O)CCOC)=O)ccc2oncc2c1 27676,C12(CNC(c3cc(C)oc3)=O)CCC(CNC(=O)C=Cc3cnc[nH]3)(CC1)CO2 27677,N1(C(C2CC2C2CC2)=O)CC2C3CCC(C2C1)N(C(C12CC(F)(C1)C2)=O)C3 27678,c1(CNC(CCC=CC)=O)nc(CNC(=O)C(C)=C2CCCC2)cc(O)n1 27679,c1(OC)cc(Br)cnc1CNc1c[nH]nc1C(N1CC(F)C(F)C1)=O 27680,N1(c2n(CCC=C)c(C3CCCC4(CCC4)O3)nn2)CCC2(C1)OCCO2 27681,c1(CC)c(C(=O)NCC2CC2CNC(C2(COC)CCCO2)=O)nnn1CC 27682,C1(C(=O)NC2C(NC(c3ccon3)=O)COC2)CC2(C1)CC(F)(F)C2 27683,c1(C(=O)NC2CCCCN(C(C3(CSC)CCC3)=O)C2)cc(N)c(C)cc1C 27684,c1(SC(C)C)ccc(C(=O)NCCOC2CN(C(=O)C(C)SC(C)C)C2)cc1 27685,C12(C(=O)NCC(c3ccsc3)C)CCC(CC1NC(=O)CC1(O)CCCOC1)C2 27686,N(C1CCCn2ccnc21)C(C1CCN(C(c2cc(CC)ncc2)=O)C1C)=O 27687,C1(NC(c2cc(O)cs2)=O)CC2CCC1(NC(C13CCC(C1)C3)=O)C2 27688,CC(C)CC(CNC(=NCc1ccsc1C(F)(F)F)NC(C)C)N1CCCC1 27689,CCCC(O)C(=O)N1CC(CNC(=O)C(C)OCCC(C)C)C1 27690,C1(C)(COC)CC(NC(=O)CCC(C)(C)F)CN1C(=O)C=C(Cl)Cl 27691,c1(C(N2CCC(NC(c3c(CC)non3)=O)C2CC)=O)cc(S(N)(=O)=O)co1 27692,c1(NCCC(C)(C)C2CC2)[nH]c(=NCC2CCCSCC2)nc2scnc12 27693,N1(C(=O)NC(c2c(C)cccc2)C)CCCCC1(C(C)C)CO 27694,C(CCN=C(NCCc1c(O)cccc1F)NC(c1ccc(Cl)c(Cl)c1)C)OC 27695,C1(C(=O)OC)CCC1S(=O)(=O)N1CCCSCC1C1CC1 27696,Cc1ccc(Cl)cc1C(=O)NC1COCCC1NC(c1cnn(C)c1F)=O 27697,C12(NC(CCCCCN(C)C)=O)CCCC1N(C(C1CCC(=O)C1)=O)CC2 27698,Cc1nn(C)c(C)c1CC(C)C(=O)NC1CCC1NC(=O)CCc1ncccn1 27699,N12CC(=O)NC(C1)C2=O.C(=O)(CC(C)C)N(CC(=O)OC)CC#C 27700,N1(C(C(C(C)C)SC)=O)Cc2ccnn2CC(NC(=O)Cc2cc(C)cs2)C1 27701,Cc1c(C)c(C)c(C(=O)NC2CCN(Cc3cn(CCCO)nn3)C2)c(C)c1C 27702,C1(SC)CC(NC(C2(C(C)NC(=O)COCCF)CC2)=O)C1 27703,C1(NC(CCSC)=O)CS(=O)(=O)N(C)C12CCN(C(=O)C1=CCCC1C)CC2 27704,CC1CN(C(=O)CC2(O)CCCCCC2)CCN1C(C1COC(=O)O1)=O 27705,C1(N(C(=O)CSSC(F)F)CC)CCN(C(C2CC2c2ccccc2)=O)C1 27706,C1(C(=O)NC(C2CCN(C(C(C)=CC3CC3)=O)C2)C)C2CCC1(C)C2(C)C 27707,N1(C(C=NOC)=O)CCOC(C(C)NC(c2csc(C(F)F)n2)=O)C1 27708,c1(CNC(=O)NC(C)C(=O)Nc2ncc(Br)cn2)ccc(CN(C)C)cc1 27709,c1(C(=O)NC2C(NC(c3cc(C4CCOC4)[nH]n3)=O)COC2)cc(O)nc(O)n1 27710,c1(CC)ccc(C(=O)NC(Cn2ccnn2)C(=O)NC(C)(C)CN(C)C)cc1 27711,c1(C(N2CC(F)(c3cn(C4CCOCC4O)nn3)C2)=O)c(O)cccc1Br 27712,C1(NC(=O)CCc2cccs2)CC2CCC1C(NC(c1ccsn1)=O)C2 27713,C1(C(C(=O)NC2CC2)N(c2ccc(OCC)cc2)C2CC2)CC2C=CC1CC2 27714,N1(C(c2c(C)c(=O)cc[nH]2)=O)CCC12CCOC(C)(C)C2 27715,Cc1nnccc1Sc1ccc(Cl)cc1.C1(c2nnnn2C)C(C)(C)N1 27716,N1(C(C(=O)NCCOC)=O)CC(NC(C2CC23CC(F)(F)C3)=O)CC(C)(C)C1 27717,C(C(C(=O)NCCc1cc(C)[nH]n1)C(C)(C)C)NC(C(CCOC)C)=O 27718,N1(C(=O)CCN2CCC(F)C2)CCC2C(CCN2C(c2cnc(O)s2)=O)C1 27719,C1(CNC(Cn2ccc(C)n2)=O)CC(NC(c2cnc(C(C)(C)C)s2)=O)CC1O 27720,C12(NC(c3cc(C)c(F)cc3)=O)CCCC1N(C(c1cc(O)nn1C)=O)CCC2 27721,N1(C(CCNC(CC(C)C)=O)=O)CC(NC(=O)COC2CS(=O)(=O)C2)CC1(C)C 27722,CC(C)CC(C(=O)NCC(C)(C)C(N)=O)N(C(=O)CN1CCC(C)C1)C 27723,N1(C(c2cc(C)n(C)n2)C(=O)NCC)CC(OC)CC(OC(C)(C)C)C1 27724,N1(C(C(C)CF)=O)CC(C2CCN(C(=O)C(C3CC3)C3CC3)CC2)C1 27725,C(=O)(CC(C)CCC(=O)N1CCOCC1CCNC(c1ncc(C)cn1)=O)OC 27726,c1(C(N(CC(C)NC(C(CC=CC)C)=O)CC)=O)ccc2nc(C)nn2c1 27727,c1(C(C)C)cc(C(N2CCC(C(C)(C)NC(c3c[nH]ccc3=O)=O)C2)=O)nn1C 27728,c1(C(N2CCC3(NC(=O)CCCCC4CC4)C(C2)C3)=O)ccc2nnc(S)n2c1 27729,C(=O)(C#CC1CCOCC1)N1CCC(NC(C(C=CC)O)=O)C1 27730,c1(C(N2C3CN(Cc4cccc(N(C)C)c4)CC32)=O)cc(O)ccc1I 27731,C1(C(=O)NC2C(NC(CCNS(CC)(=O)=O)=O)CCC2)CC(=O)OC1(C)C 27732,c1(NCC(O)COC(C(CC)(C)C)C)ccc(C(N)=O)c([N+](=O)[O-])c1 27733,n1(CC(=O)NC(CCNC(CC(C=C)CC)=O)C)ccc(=O)n(C)c1=O 27734,N1(C(c2cc(OC)n[nH]2)=O)CC(C(=O)NC23CC(F)(C2)C3)C2(CCC2)C1 27735,N1(C(COC)C)CCC(C)C(NC(C2CCCCC2c2ccccc2)=O)C1 27736,Cc1ccc(C(C)NC(CC(N)=O)C2CCOCC2)nn1 27737,c1(C(=O)NC(C)CN(C(=O)C(F)n2ccnc2)C)cnc2c(c1)NC(=O)CO2 27738,N1(C(CC)=O)CCOCC(CNC(=O)CC2CCCN2C(C)=O)C1 27739,c1(-n2c(-c3c(C)ccnn3)nc(C3CCOCC3)n2)ccc(F)c(Br)c1 27740,C(CCNC(c1cccc(F)c1)=O)(C(F)(F)F)NC(C)C(=O)NC(C)(C)C 27741,C1(C(=O)Nc2cnn(-c3ccc(OC(F)F)cc3)c2)CCCN(CC(F)F)C1 27742,C(=O)(C1COc2ccc(F)cc21)N1CC2(CCN(C(C(CC=C)CC)=O)C2)C1 27743,C1(CN(C)C(C2CCCN2C=O)=O)COCCN1C(=O)C(F)=C1CCCC1 27744,C1(C(=O)NC2C3CCCOC23)COCCN(C(c2ccc(C3CC3)o2)=O)C1 27745,Cc1cc(C(=O)NC2CC(NC(=O)C=C3CCCCC3)C2)nnc1C 27746,C(=O)(C(CC)C(C)C)NC1(CCNC(c2c(CC)cc[nH]2)=O)CC1 27747,C1(NC(C2CC(C)(CC)C2)=O)CCN(C(=O)CCOCC(C)(C)C)CC1 27748,c1(OC)ccc(C(=O)NC2(C)CCCN(C(C3(CCN(C)C)CC3)=O)C2)cc1Cl 27749,N1(C(C(CC)CO)=O)CCN(C(C2CC(=O)NC2(C)C)=O)C(C)C1 27750,N1(C(C2CC3C=CC2C3)=O)CCC2(CCC2)C(NC(C2(C3CCC3)CC2)=O)C1 27751,N1(C(C2N(C(C(CC)N(C)C)=O)CCC2CC)=O)CCC2C(O)CC12 27752,c1(C(=O)NCC2CCC(C(N3CC4(CCOC4)C3)=O)CC2)nccc2cc[nH]c12 27753,c1(C(=O)NCCC2CCCN(C(=O)C(O)C3CC3)CC2)c[nH]c2cccc(Cl)c12 27754,C12(NC(c3ccc(CC)nc3)=O)CCCC(CN(C(=O)C(Cl)=CCl)C1)C2 27755,CC(C)(C)CC(=O)N1CC(O)CC1C(=O)NC(CO)C(N)=O 27756,C(=O)(C(C)S(C)(=O)=O)N1C(C(C)NC(=O)C=Cc2cc(C(N)=O)co2)CCC1 27757,c1(C(=O)NC2CC(N(C(=O)CC3CCCO3)C)C2)cnc2c(c1)CCOC2 27758,C(=O)(C(C)CC(C)(C)C)NCc1ccc(CN(C(c2onc(C)c2C)=O)C)cc1 27759,c1(CC(=O)NCCCNC(C2(c3ccccc3)CC2)=O)cncc(F)c1 27760,C1(O)(CN(C)C(c2ccc(Cl)cn2)=O)CCN(C(C2CCC(CCO)CC2)=O)C1 27761,N1(c2ncnc3n[nH]c(C)c32)CCC2CC(CNC(=O)C=CI)CCC2C1 27762,Cc1cncc(CC(=O)NC2(CC(=O)NC3CCSCC3)CCCCC2)c1 27763,c1(C(N2CC=CC(NC(C#CC(C)C)=O)C2)=O)cccc2c1COC2 27764,C1(C(=O)NC2CCCC(CC(=O)NCC3C(C)(C)COC3)C2)CCC2(CCC2)C1 27765,C(=O)(CC1=CCOCC1)N(CCCC(=O)NC1CCNC1=O)C 27766,C(CC)(C(=O)NCC(O)CNC(C1(n2cccn2)CCC1)=O)OCC 27767,c1(SC)cc(C(=O)NC(C)CN(C)C(C2(c3ccccc3)CCCC2)=O)c(C)o1 27768,N1(C(c2scc(C)n2)=O)CCC(F)(CNC(C2CC2(Cl)Cl)=O)CC1 27769,CC1CN(C(=O)CC2CCC(C(N)=O)CC2)CCN1C(=O)COc1cnn(C)c1 27770,C=CCCC(C(=O)NOC(CO)C(C)C)NC(=O)C(=O)C(C)(C)C 27771,c1(C(=O)NCCC2N(C(Cc3nnc(C)o3)=O)CCSC2)cnn2cnnc2c1 27772,c1(C(=O)NC(C(C)NC(C2CNC(=O)C2)=O)CO)cnc2nccn2c1 27773,c1(C(=O)NCC=CCNC(c2ccc(F)cc2C2CC2)=O)cc(F)c(O)c(Cl)c1 27774,C12(NC(C3Cc4ccc(F)cc4C3)=O)COCCC1CN(C(c1ccsc1)=O)C2 27775,CC1(NC(C2CC3(C2)CC3F)=O)CCN(C(=O)C(c2ccccc2)C2CC2)CC1 27776,c1(C(N2CC(NC(c3c(C)ccc(F)c3)=O)C(C)C2)=O)ccc2[nH][nH]c(=N)c2c1 27777,C1(NC(c2cc(C)[nH]n2)=O)CCCC(N(C(=O)C(F)=CC2CC2)C)C1 27778,C1(NC(c2noc(CC)c2C)=O)CN(C(c2c(C)noc2N)=O)CC1S(C)(=O)=O 27779,C(=O)(C1CSc2ccccc21)N(C)CC1CCN(C(c2ccnn(C)c2=O)=O)C1 27780,Cc1cc(NC(C2CCCN(C(=O)CCCF)CC2)=O)cc(Cl)c1 27781,c1(C(N2C(C(=O)NCCSCCC=C)CCC2)=O)cccc(=O)o1 27782,N12Cc3n[nH]cc3C1C(=O)C(=O)C2c1cn(CCNC(C)=O)nn1.CN.OC 27783,N1(C(CCNC)=O)CC(C2CCCCC2)C1.CC(O)C(C)(C)C.c1(=O)ccc1=O 27784,C1(C(N2CCC(C(C)C(=O)NCc3ccc(OC)o3)C2)=O)(OCC)CCOC1 27785,c1(CC)ccc(NC(=O)CC2CCCN(C(=O)C(C#N)=CC3CC3)C2)cc1 27786,c1(CC)c(C(=O)NC(C)CCNC(C2CCOC2)=O)nnn1CC 27787,C1(C(=O)NCc2cc(C(=O)NCC(C)C3CC3)no2)(CC)CCCCC1 27788,c1(C(=O)NC(c2cc(Br)ncc2F)C)cc2n(n1)CC1(CC1)CO2 27789,C1(N(C(COC)=O)C)CCCN(C(C2CCCS2(=O)=O)=O)CC1 27790,c1(C(=O)NC2CN(C(C3(C)CC3(F)Cl)=O)C2)cccc(NC(N)=O)c1 27791,C1(CC(C)NC(c2cccnn2)=O)CCN(C(C2CNC(=O)C2)=O)CC1 27792,C(C)(C)(C(C)(C)O)NC(C1C(CNC(c2c(OC)scc2)=O)C1(C)C)=O 27793,C1(C(=O)NC2CC3CN(C(C=CC(=O)NC4CC4)=O)C2C3)CCn2nncc2C1 27794,C=C(CNC(C1(C)C=CCN1C(C12CC(F)(C1)C2)=O)=O)C1CCOCC1 27795,C1(C(=O)OCC)(NC(=O)NC2CC2(c2ccc(Br)cc2)C)CCOCC1 27796,N1(CC(=O)NC2CN(C(C(C)OCCC(C)C)=O)C(C)C2)CCc2ccccc21 27797,c1(C(COC)(C2CC2)NC(c2ccc(Cl)s2)CC)nnnn1CCN1CCCC1=O 27798,C1(C(N(CC#C)CCOC)=O)(NC(=O)Cc2ccccn2)CC1(C)C 27799,N1(C(c2cnc(OC)s2)=O)CCN(C(C2CC(=O)NC2(C)C)=O)C(C2CCC2)C1 27800,C1(C(=O)NCC(N2CC=CC2)C)CSCCN1C(=O)C(=O)NCC(F)F 27801,c1(C(=O)NCC(CC)N(C)C(c2scnc2Cl)=O)cn(C2CCC2)nn1 27802,N1(C(C(CCC)(C)CCC)=O)CCC2(CC1)CC(NC(C1CC(C)C1)=O)CCO2 27803,C(=O)(C(CC=C)CC(C)C)NC(CC#C)(C)C(=O)NCCC1CCCC12CC2 27804,CC1(C)CC(CNC(=O)CC2CS(=O)(=O)C2)N(C(=O)C=Cc2cccc(Cl)c2)C1 27805,C1(NC(C2=NOC(C)C2)=O)CC1C1CCCN(C(C23CC(C2)C(C)(C)O3)=O)C1 27806,N1(C(C2(OC)CCSC2)=O)CC(C)CN(C(c2cccc(=O)n2O)=O)C(C)C1 27807,N1(C(=O)CCC2CCOC2)CC2CC1CN2C(C1C2(CC2)C12CC2)=O 27808,c1(C(N2CCC(C)(NC(C(CC=C)C)=O)C2)=O)c(C)ccc2ncccc12 27809,C1(SCC(=O)NC2(C)CC(NC(C3CCSCC3)=O)C2)CCS(=O)(=O)C1 27810,c1(C(N2CC3CC(NC(c4c(O)cc(C)nn4)=O)C3C2)=O)ccc(C#N)nc1C 27811,C1(CSC)CCCN1C(C1CCOC1CNC(=O)CCCC1CCC1)=O 27812,N1(C(c2c(OC)c(F)ccc2)=O)CCC2CN(C(=O)CCCN(C)C)CC12 27813,c1(C(=O)NCc2ncoc2C2CC2)ccc(C(F)(F)F)c([N+](=O)[O-])c1 27814,C1(C2CCN(CC(F)(F)F)CC2)(c2c(Cl)ccc(=N)[nH]2)CC1 27815,C(=O)(C1=C(Cl)CCC1)NC(C(=O)N(C)CCc1cccs1)CCF 27816,c1(OC)cc(F)c(F)cc1C(=O)NC1CC(C(=O)NCc2ocnc2C)C1 27817,N1(C(C(C(=O)OC)OC)=O)CC(F)(F)CC1CCNC(C1CCCN1C(C)C)=O 27818,C#CC1CN(C(=O)CC2C(CC)C2(F)F)CCN1C(c1cc(Cl)cs1)=O 27819,C1(C(=O)NCC(CNC(C2(CC3CC3)CCC2)=O)O)CCNC1=O 27820,C(=O)(C(C)(C)C(C)O)Nc1cccc(-c2cn(C(C)C(=O)O)nn2)c1 27821,C(=O)(C(C(C)NC(c1cccn1C)=O)C(C)C)Nc1c(C)noc1 27822,c1(CNC(C2CNCCN2Cc2ccc(Br)c(Cl)n2)=O)ccc(O)c(O)c1O 27823,CN1C(=O)NC2(CCC(C(=O)N(c3ccncc3)C)CC2)C1=O 27824,C(=O)(C(CC)CC(F)(F)F)NCC(C1CC1)NC(c1c(C=C)cnn1C)=O 27825,c1(OC)ccc(C)nc1C(=O)NCC(c1ccccc1)NC(=O)C(C)C(C)(C)O 27826,c1(N2CCC(CCNC(c3ccc(CC)[nH]3)=O)CC2)nc(O)c2ccccc2n1 27827,CC1CC(CNC(=O)CC2(O)CCOC2)CN1C(=O)C(c1ccc(F)cc1)=O 27828,c1(NCc2c(C)cccn2)ncc(S(=O)(=O)NCC2CC2C)cc1Cl 27829,CC1(C)CC(=O)OC1CNC(=O)CC1CC(NC(C2C3CC4C(C3)C24)=O)C1 27830,Cc1ncnc(NC2CC(CNC(c3cnc(Cl)s3)=O)C2)c1Br 27831,C1(C(=O)NCC2CC2Cl)(CNC(=O)CC2CC3CC3C2)CC12CCC2 27832,Cc1[nH]c2ccccc2c1CC(=O)NCC1(O)CCN(C(=O)COC(F)F)CC1 27833,c1(C(=O)OC)c(F)cc(CNCCCc2cncnc2)cc1F 27834,c1(C(C)OCCN(C)C)nc(-c2ccoc2)nn1C1CCOC1(C)C 27835,C1(CSCC(=O)NC(C)CC2CN(C(C3CC(F)C3)=O)C2)CCCCO1 27836,c1(C(N2C3CC(CNC(C4(CC)COC4)=O)(OC3)C2)=O)cc(OC)c(N)c(N)c1 27837,C1(CC(=O)NCCC2(NC(CSC(C)C)=O)CCCC2)CCC12CCC2 27838,Cc1[nH]nc(CO)c1C(N1CCC(CCC(=O)N(C2CCCC2C)C)C1)=O 27839,c1(CC)nn(C)c(CC(=O)NCCCC(C)NC(=O)C(C)C(F)(F)F)c1Cl 27840,Cc1cc(NC(=O)NCC2CCSC2(C)C)cc(C(F)(F)F)c1 27841,n1(CCC)ccc(C(C(=O)NCC2CC2)N(CC(c2ccccc2)(F)F)C)n1 27842,Cc1c(C(N2CCC(N(C(=O)Cc3cnoc3)C)C2)=O)oc2c(C)cccc12 27843,CON1CCC(C(=O)NC2CCC(C)N(C(=O)CCc3ccc(Cl)s3)C2)CC1 27844,CCCC(C)C(=O)NC1CC(C)(NC(=O)CCc2ccccn2)C1 27845,C1(O)(C(=O)NCC2(O)CN(C(CCc3cnc(C)o3)=O)C2)CCCC(C)CC1 27846,C1(C(=O)NCC(C(C)C)NC(C(C(=O)NC)(C)C)=O)CCc2nc(C)ncc2C1 27847,C(=O)(C(=O)C(C)(C)C)N1CC(C(=O)NCCC(C)C)C(F)C1 27848,C1(O)(CN(C)C(c2cnns2)=O)CN(C(=O)CCN2CCC2)C1 27849,C1(C(=O)NC2CCC(NC(C(OC)OC)=O)CC2)CC(F)(F)CCC1(C)C 27850,N1(C(C(COCC)C)=O)CC(CC(=O)NCCn2cc(C)cn2)CC1(C)C 27851,c1(C(N(C2CCN(C(C(COC)(C)OC)=O)C2)CCO)=O)cncc(F)c1Cl 27852,c1(C(N2CC(CC)N(C(=O)CCn3cc(Cl)cn3)CC2)=O)ccnc2ccsc12 27853,c1(C(N2CCCC(Cn3cc(C(COC)(C)O)nn3)C2)=O)cncc(F)c1Cl 27854,c1(CCCC(=O)NC23C(CN(C(CC(=C)C)=O)C2)C3)csc2ccccc12 27855,c1(C2(O)CN(CC(=O)NC(C(C)(C)ONC(=O)OC(C)(C)C)=O)C2)ccc(Cl)nc1 27856,Cc1nc(C(=O)N(CC)CC2CCCN2C(=O)CC2CCCN(C)C2)cc(O)n1 27857,Cc1cc(C(=O)NC2CCN(C(=O)CCC3CN(C(=O)OC(C)(C)C)C3)C2)cs1 27858,C(=O)(C#CC1CC1)NC(CC)CN(C(C1CCCN(C(C)C)C1)=O)CC 27859,c1(OC)cnc(C(=O)NCCCNC(c2sccc2-n2ccnn2)=O)c(OC)n1 27860,c1(-c2cn(CC(CNC(c3ccc(CCC)[nH]3)=O)OC)nn2)c(F)cccc1F 27861,C#CCCC(C(=O)NC12CCC(CC1)CC2)NC(=O)CN(C(=O)COC)C 27862,C(CC)(CC)(CCNC(=O)C(C)S(N)(=O)=O)NC(CCN(C(CC)CC)C)=O 27863,c1(C(=O)NCC(CN(C(C(C)C(F)(F)F)=O)C)O)cccc2c1N(C)C(=O)CO2 27864,O=[N+]([O-])c1ccc(N2CCC(COCC(F)(F)F)C2)c2ccncc12 27865,CC(C)C#CC(=O)N(CC(C)NC(c1cnn(C(C)C)c1Cl)=O)C 27866,CC1(C)CN(C(=O)CCCNC(C2(C)CCC(=O)NC2)=O)CC1O 27867,C(CN=[N+]=[N-])(C(=O)NC12CCC(CC1)CC2)NC(CC=C)=O 27868,OC1CCCCC(NC(C23CCC(CC2)C3)c2nnnn2C2CCCC2)CC1 27869,N1(C(c2cc(C(C)=O)sc2)=O)CCCCC1CN(C)C(c1csc(F)c1)=O 27870,C1(C2CCN(c3ncnc4c3CCC4)CC2)(NC(=O)CC2NC(=O)NC2=O)CC1 27871,N1(C(COCC#C)=O)CCCC1CN(C(C1(C#C)CC1)=O)C1CC1 27872,CC1CCC(C)(C(N2CC3CC2(C(=O)NCC(O)CN(C)C)C3)=O)CC1 27873,c1(CNC(CCN(C(C2CCN(C)C2=O)=O)CC)=O)cncc(OC)c1 27874,CC1(C)C(C(=O)NCC(C)(F)CNC(=O)CCNC(=O)CO)CC1(F)F 27875,CC1=NC(C)(CNC(c2coc(C(C)NC(c3cnc(C)o3)=O)n2)=O)CS1 27876,C(=O)(CC(C(F)(F)F)NC(c1[nH]ccc(=O)c1C)=O)N(C(C(CC)C)C)C1CC1 27877,C(=O)(C(CC(=O)OC1CC1)N(C)C)NC(C(C)NC(C=CC=CCC)=O)(C)C 27878,c1(OC)cc(F)cnc1NC(C1CCN(Cc2ccc(C)s2)CC1)=O 27879,C1(NC(c2cc(CO)on2)=O)CN(C(c2c[nH]nc2C2CC2)=O)CCC12CCC2 27880,C1(C(=O)NC2CC3CN(C(CP(C)(C)=O)=O)C(C2)C3)CCC(S(N)(=O)=O)CC1 27881,n1(CC=C)cc(CNC(=O)C(F)CC2CN(C(=O)CSC(C)C)C2)nn1 27882,CCC(C)C(C(=O)NCc1cc(C)ncn1)NC(C1C2CCC(F)C12)=O 27883,c1(SC)ncc(C#N)c(N2CCN(c3ccnc(Br)n3)C3CC23)n1 27884,c1(C(N2CCCN(C(Cc3c(C)nsc3)=O)CC2C)=O)cccc2c1OCC2C 27885,N1(C(c2n(CC)ncn2)=O)CCCN(C(c2cc(C#N)oc2C)=O)CC1CO 27886,c1(C(=O)NCC2CCCC(NC(CC(=O)N(C)C)=O)C2)cc(N)ccc1Br 27887,C(F)(C(=O)NN1CCCC1C(=O)NC(C1CCCOC1)(C)C)=C(C)C 27888,CCC(C)CCCCC(=O)N1CCC(NC(C2(CO)CCC2)=O)CC1 27889,S(=O)(=O)(c1ccc(CCC(=O)NS(=O)(=O)C(Cl)(Cl)Cl)cc1)NC1CCC(OC)C1 27890,N1(CC)CCC1C(=O)NC1(CC(=O)NC2(c3cc[nH]n3)CC2)CC1 27891,c1(C(=O)NC(C2N(C(C(C)=C3CCCC3)=O)CCC2)C)cn2c(n1)C(C)CCC2 27892,C1(NC(C2CC2c2ccncc2Cl)=O)CCCN(C(C2(F)CC=CC2)=O)CC1 27893,C=CCC(CNC(=O)COC(C)(C)CC)C(=O)NC(C)CN1CCCC1 27894,C1(C(=O)NC2CC(C)(NC(c3ccc(CC)o3)=O)C2)CCOC1(C)C 27895,c1(OC)ccc2c(=NC(C)CSC(F)F)[nH]c(=NC3CCCN(C)C3)[nH]c2c1 27896,C(CNC(=O)C(C)(C)F)(CCNC(=O)CCc1cc(C)no1)OC 27897,Cc1nc2c([nH]1)CC(C(N1CCC3CN(C(=O)C(=O)NC4CC4)C3C1)=O)CC2 27898,Nc1cc(O)nc(O)c1C(N1CCC(O)(c2cccc(C(F)(F)F)c2)C1)=O 27899,CCS(=O)(=O)CC(=O)N1CC(C(N2C3CCCC2CC3)=O)CC1(C)C 27900,c1(C(=O)NCCOCCN(C(=O)Cc2ccoc2)C)c(Cl)ccc(F)c1N 27901,C1(C(N2C(C)CN(C(c3ncccc3N(C)C)=O)CC2)=O)CCCCN(C)C1=O 27902,Cc1ccc(N(C(c2ccc(C(c3cc(Br)ccn3)=O)cc2)=O)CC2CC2)cc1 27903,C1(CNC(c2cn(CC)nc2)=O)C2CN(CC(=O)Nc3cncc(Cl)n3)CC12 27904,CCC(CC(=O)N1C2CCC1CC(CNC(=O)CCCS(N)(=O)=O)C2)C(C)C 27905,N1(C(c2nc(C(C)OC)sc2)=O)CC2(CC(NC(c3cc(C)sc3C)=O)C2)C1 27906,N1(C(C(CC)n2ccnc2)=O)CCC2(CC1)CC2NC(c1cnc(COC)s1)=O 27907,CC(CS(C)=O)C(=O)NCCCCN1CCCN(C(=O)CCN(C)CCO)CC1 27908,c1(C(N2CCC(NC(CCCNC(C)=O)=O)C2)=O)cccc(C)c1N 27909,C1(C)(C(=O)NC(C2(CN3CCCC3)CC2)C)CCCN1C(=O)CN1CCCCC1C 27910,N1(C(c2ccc(CNC(C(CCC=C)(C)C)=O)cn2)=O)CCc2c(O)noc2C1 27911,Cc1ccc(O)cc1C(=O)NC(C)C(c1ccccc1)NC(=O)CSC1CC1 27912,C(CC(C)(C)C(=O)NCC1CN(C(C2CCC(C)CC2)=O)C1)SC 27913,C(C(=O)NCCc1c[nH]nc1O)(C(C)(C)O)NC(c1c(CC)n(C)cc1)=O 27914,C1(C(N(c2c(C)csc2)C)=O)CC12CC2(F)F 27915,C1(OC)CC(CNC(c2ncc(F)cn2)=O)N(C(c2cnc(C(C)(C)C)o2)=O)C1 27916,c1(C(N2CCCC(NC(CC(=C)C)=O)CC2)=O)c(F)ccc(O)c1F 27917,C1(C(=O)NC(C)C2CC2)CC12CCN(Cc1noc(C(F)(F)F)n1)CC2 27918,N1(C(COC(CC)(C)C)=O)Cc2cccc(CNC(=O)CC3CCC4CC34)c2C1 27919,C(CC(C)C(=O)NCCN(C(=O)C(c1cnn(C)c1)=O)CC)=CCC 27920,Cc1nc(Cc2ccc(F)cc2)oc1C(=O)NCC1CCN1C(C1CN(C)C1)=O 27921,S(=O)(=O)(c1ccc(OC)c(-c2ccc(OC)cc2CC)c1)N(CC#C)C(C)C 27922,N1(C(c2ccn(COC)n2)=O)CCC(C)C(NC(=O)C(C)(O)C2CC2)C1 27923,C1(N(C(CCOCCC)=O)C)CN(C(=O)Cn2c(C)c(C)sc2=O)CC1(C)C 27924,C1(N(C(=O)CC2(C(N3CCC3)=O)CC2)OC(=O)C2CC2)CCNC(=O)C1 27925,C1(C(=O)NCc2cc(C(N)=O)no2)CCCN(C(C2CC3CC2CC3O)=O)CC1 27926,c1(CC)ccc(S(C)(=O)=O)cc1C(=O)NC1C2CC3CN(C(=O)C4CC4)C1C3C2 27927,c1(OCC(=O)NC(C2CCCN2C(=O)COc2ccon2)C)cc(F)cc(F)c1 27928,C1(OC)(NC2CCC(n3cc(CCC(C)(C)CO)nn3)CC2)CC(C)(C)C1 27929,c1(CNC(c2cccc(CN3CCCC3=O)c2)=O)ccc2c(c1F)OCCO2 27930,c1(N2CCC(CCN(CCCCCOCC)CCO)CC2)ncnc2scc(Br)c12 27931,N1(C(=O)NCCC(=O)OC(C)(C)C)CCC2(CCCCC2)CC1 27932,C(=O)(CCCCc1ccccc1)N(C1CCC(NC(c2cncc(O)c2)=O)C1)C 27933,c1(C(N(C2CN(C(c3cccn3C)=O)CC2F)C)=O)ccc2cc(F)ccc2n1 27934,N1(C(C2C(C(C)C)OCC2)=O)CC2(CC(C(=O)NCCC(=O)N3CCCC3)C2)C1 27935,C1(OC(C)=O)(NCc2cc(F)ccc2Cl)CCC(C(F)F)CC1 27936,c1(NCC2CCC(NC(c3c(CC)nco3)=O)C2)ncccc1C#N 27937,C1(CC(=O)NCC(CNC(C2(CC(C)C)CC2)=O)OC)CC2(C1)CC1(CCC1)C2 27938,Cc1nnc2n1CC(c1nc(C3CC=CCC3)nn1-c1nccn1C)CC2 27939,c1(C(=O)NCCC2(OC)CN(C(C3CCCC3C)=O)C2)c(C)nn(C(C)C)c1C 27940,C1(NC(C2CC3(C2)CC(O)C3)=O)CCN(C(=O)C(F)(F)C(O)C2CC2)CC(O)C1 27941,C1(NC(CCc2cnc(C)s2)=O)CCN(CCC2CCOC2)CC1(C)C 27942,c1(C(=O)NC2(c3cccc(F)c3)CCN(C(C(C=C)O)=O)C2)ccc(N)c(Cl)n1 27943,C1(F)(CNC(c2c(CCC)nco2)=O)CCC(NC(c2ccoc2Cl)=O)C1 27944,C1(O)(CNC(C(C)OCCOCC)=O)CCN(C(c2scc(C)c2C)=O)C1 27945,c1(C(=O)NCC(CNC(c2[nH]nnc2-c2ccnn2C)=O)OC)cocc1C 27946,c1(SCC)nccnc1C(N1CC(OC)CC1CCNC(C1CC(C)(C)C1)=O)=O 27947,O=C1CCc2ccc(C(=O)NC3CCCC(NC(c4n[nH]cc4Cl)=O)C3)cc2N1 27948,c1(OC)ccnc(C(=O)NC2CC(C(=O)O)(SC)C2)c1C 27949,C(C(=O)N1CC(N2CCOC2=O)C1)(C(C)(C)C)NC(c1c(C)ccnc1)=O 27950,C1(CC(=O)NC(C)C(C)NC(=O)Cc2ccoc2)C2CC3CC(C2)CC1C3 27951,N1(Cc2c(C#N)c(F)ccc2)CCC2(CC1)CCN2C(c1cc[n+]([O-])cc1)=O 27952,c1(CCC)[nH]nc(C(=O)NCC2CCN(C(C3CC3C)=O)C2(C)C)c1[N+](=O)[O-] 27953,N1(C(C2(SC)CCC2)=O)CC2CCC(NC(=O)C=Cc3ccc(C)s3)CC2C1 27954,C=CCCCC(=O)NCCC1CN(C(=O)CCN(C(C)CCC)C)CCO1 27955,N#Cc1cc(C(=O)NCC(C2CCCC2)NC(c2ccn(C3CCC3)n2)=O)c[nH]1 27956,N1(C(C2(C#C)CN(C(c3cn(CC)cn3)=O)C2)=O)CCOC(CC)CC1 27957,O=C(O)CCCn1cc(C2(O)CN(C(=O)CCN3CCOCC3)C2)nn1 27958,N1(CC2(NC(C3CCN(C4COC4)C3)=O)CCCCC2)CCC(F)(F)CC1 27959,C1(N(C)C(c2ccc(Cl)cn2)=O)CCCC(NC(=O)CSc2nnnn2C)C1 27960,C1(C(=O)NC(CC(C)NC(C(C)S(N)(=O)=O)=O)C)CN(C)CCN(C)C1 27961,N1(C(C2CCC(CCCCC)O2)=O)CCN(C(c2ccc(C)cc2)=O)C(C)C1 27962,C1(OC)CC(CNC(=O)CNC(c2ccoc2)=O)N(C(c2cnc(C)[nH]2)=O)C1 27963,C1(CNC(C2(COC)CCCC2)=O)CCN(C(c2cccs2)=O)C12CC2 27964,Cc1ccc(F)c(C(=O)NCC2CC(C(=O)NCC(c3cnn(C)c3)C)=NO2)n1 27965,C1(C(=O)NC2C(CNC(c3cnn(CC)c3C)=O)CCC2)CC12CCCCCC2 27966,N1(C(C2CCCC2O)C(=O)NC(=O)NCC)CC(N(C)C)Cc2ccccc21 27967,N#Cc1ccc(CC(=O)NC2CCN(C(=O)CSc3nncs3)CC2F)cc1 27968,c1(C(=O)NC(CCS(C)=O)CNC(=O)C#CC2(C)COC2)nc2ccccc2[nH]c1=O 27969,CC1(C)CCN(CC(=O)NCC(C)(O)CNC(c2cc(C#N)c[nH]2)=O)C1 27970,Cc1ccc(C(F)CN)cc1C.C1(c2ccccc2)CC(=O)N1C(C)C(C)C 27971,C1(CCC(=O)NC2(CNC(c3cc(C(C)=O)sc3)=O)CC2)CCCCN1C 27972,C1(NC(Cc2c(CC)con2)=O)C2CC(NC(C3(C)CCSCC3)=O)CC12 27973,Oc1nc(C23CCCCC2C3)nc2c1CNCC2 27974,N1(C(c2nc(CC)oc2)=O)CCN(C(=O)CN2CCC(CC(=O)OC(C)(C)C)CC2)CC1 27975,C#CCCCCC(=O)NCC12CC1CN(C(c1ccc(C)cc1)=O)C2 27976,c1(CNC(C2CCCN(c3ccncn3)C2)=O)ccc(C(=O)O)c(F)c1 27977,CC(C)(C)C(C#N)C(=O)N1CCC(O)(CNC(c2cccc3nc[nH]c23)=O)CC1 27978,C1(C)(COC)CC(NC(c2n[nH]c3c2COC3)=O)CN1C(c1cc(Cl)cn1C)=O 27979,C(=O)(C(C(C)(C)O)NC(=O)C(C)n1cccc1)NC(c1ncc(C)cn1)C 27980,C1(CCNC(c2n(C=C)ncc2)=O)CC2CCC(C1)N2C(C1CCN(C)C1C)=O 27981,c1(C(N2CCC(C(C)(C)NC(C3OCCCO3)=O)C2)=O)cn2c(n1)CCC2 27982,c1(CC)cc(C(=O)NCC2(C(N)=O)CN(C(=O)COCC(F)F)C2)cc(Cl)n1 27983,c1(C(N(CC(C)O)CCNC(c2cccc[n+]2[O-])=O)=O)cnc2ncccc2c1 27984,C(=O)(C1CCc2snnc21)N1C2CN(C(CN(S(C)(=O)=O)C)=O)CC1CC2 27985,O=C1CCCC(C(=O)NCC(N2CCN(C(=O)CCn3cncn3)CC2)=O)O1 27986,Cc1ccc(CC(=O)NC(C)CCCNC(C2C=CCC2)=O)c(C)c1 27987,CCCCCCNC(=O)C(Cc1cnc[nH]1)NC(=O)CSc1cn[nH]c1 27988,c1(C(N2CCC(CNC(=O)C(F)(F)C3CC3)C(O)C2)=O)ccc2ncnn2n1 27989,N1(C(c2c(CC)nco2)=O)C2CCC1CN(C(=O)Cc1noc(C)n1)C2 27990,Cc1cnc(Cl)c(C(N2CCC(CC(C)NC(c3ccc(F)nc3)=O)CC2)=O)c1 27991,c1(C(=O)NCC2OCCN(C(CS(CC)(=O)=O)=O)C2)ccc(OC)c([N+](=O)[O-])c1 27992,C(N=c1[nH]c(C)c(C(=O)NC(CCO)C(C)C)s1)c1c(F)ccc(OC)c1 27993,Cc1cc(NC(=O)C(=O)N(C)Cc2ccnc(Cl)c2)cnc1C 27994,c1(C(=O)NCC(Cc2ccccc2)CO)csc(=NCc2ccc(O)c(Cl)c2)[nH]1 27995,Cc1cc(C(F)F)oc1C(=O)NC(C)CC(C)NC(c1ccncn1)=O 27996,Cc1ccc(C(=O)NCC2CN(C(c3nnn(C)n3)=O)CC2C)c2ccccc12 27997,c1(CC)ccc(OCC(N2CCC(C)C2CNC(C2(O)CCSCC2)=O)=O)cc1 27998,N1(C(CCn2ncn(C)c2=O)=O)CC2CC(NC(c3cnccc3Cl)=O)C2C1 27999,C1(NC(CCC=CC)=O)CC2CC(NC(c3cc(OC)cnc3F)=O)CC2C1 28000,N1(C(C(C2CCCC2)SC)=O)CC(F)(C(=O)NOCCOc2ccncc2)C1 28001,c1(C(N2CC(COC)(CNC(=O)C(C)(Cl)Cl)C2)=O)ccnc(S(N)(=O)=O)c1 28002,C12(CNC(c3c(CC=C)cccc3)=O)CN(C(=O)CN=S(C)(C)=O)CC1CCO2 28003,CC1CN(C(C2(C(C)NC(c3ccccn3)=O)CC2)=O)CC(CO)O1 28004,N1(C(C(C(C)C)C2CCC2)=O)CCC2(C=C(C(=O)NC34CCN(CC3)C4)C2)C1 28005,C1(CN(CCC(CC)C)CCOC)COc2ccccc2O1 28006,c1(NC2(CCC)CCN(C(=O)C(C)(CC)OC)CC2)cccc(CO)c1[N+](=O)[O-] 28007,Cc1ccc(-n2nccc2C)c(NC(C2CCN(Cc3ccsc3)CC2)=O)c1 28008,C1(NC(c2ccc(C#C)o2)=O)CCN(C(=O)C(C)(C)c2ccnn2C)CC1C 28009,N1(C(C(CSC)(C)C)=O)CCOC2(C1)CN(C(=O)CCc1cccnc1)C2 28010,C1(NC(CN(C(C)C)C)=O)CC(O)CN(C(=O)CN2CCC(O)CC2)C1 28011,Cc1nnc2n1CC(C(N1CC3CCN(C(=O)C#CC(C)(C)C)C3C1)=O)CC2 28012,N1(C(c2cnc(N(C)C)o2)=O)CCC2C1CCN2C(c1ccc(=O)oc1)=O 28013,C1(C(=O)N)CN(C(c2c(C)nc(-c3ccccc3)s2)=O)CC(F)(F)C1.C(C)C1CC1 28014,N1(C(C(=O)NCc2cc(OC)c(C)cc2)=O)CC2CCC(C1)C(=O)N2 28015,c1(CNC(N(C2CC(F)(F)C2)CC)=O)c(C(F)(F)F)coc1C 28016,c1(C(N2CC(C)C(F)(F)C2)C(=O)NCCCSCC)ccc(C#N)c(C)c1 28017,C1(NC(C2(SC)CN(C(=O)C=CC3CCC3)C2)=O)CCOC(C)(C)C1 28018,c1(CC(=O)NC(CNC(C(CCC)(C)O)=O)(C)C)ccc(S(C)=O)cc1 28019,C1(NC(CN(C(=O)Cc2c[nH]nc2C)CC#C)=O)CCCCC1N(C)C 28020,N1(C(C(C)NS(C)(=O)=O)=O)CC2C(N(C(=O)CNC(N3CCOCC3)=O)C)C2C1 28021,N1(CCCNS(CC)(=O)=O)CCC(C(=O)NCc2cc(C(C)C)no2)C1 28022,C1(CCCNC(CCNC(=O)Cn2cc(CO)nn2)=O)(CO)CCOCC1 28023,N1(C(c2ccc(CC)cc2C)=O)CC(C)N(C(c2cnc(S)n2C)=O)CC1C 28024,C1(NC(CC(C)n2ccnc2)=O)C2CC3CN(C(=O)Cc4cnsc4)C1C3C2 28025,Cc1oc([N+](=O)[O-])cc1C(N1CC2CC1CC2CNC(=O)CCC1CC1(Cl)Cl)=O 28026,c1(C(=O)N(CC(CO)NC(CC2C(CC)C2)=O)CC)ccc2ccccc2n1 28027,Cc1occc1C(=O)NC1CCC1C(=O)NCCNC(=O)N(C)C 28028,N1(C(C(CCC)O)=O)CC(NC(c2cccn2C)=O)CC12CCCCC2 28029,Cc1c(C(=O)NCC2(F)CC(NC(=O)CN3CC4CCC3C4)C2)nnn1C 28030,CC1CCN(C(=O)CCN2CCCC2)C(C(=O)NC2CC3CC4C(C3)C24)C1 28031,C1(CC(=O)NC2(CNC(Cc3ccc(C)s3)=O)CCCC2)CCCCC1O 28032,c1(C(N(CCC(C)NC(C2CCCC2(C)C)=O)C)=O)cnc(N)c(Br)c1 28033,O=C(C(O)C(F)(F)F)N1CCN(C2CN(C(C3(Cl)CC3(F)F)=O)C2)CC1 28034,N1(C(C(CCC)OC)=O)CCCC(F)(C(=O)NC2CC2CC(C)(C)C)C1 28035,c1(C(N(C(CCNC(CN(CC)CC)=O)C)C)=O)cc(C(=O)OC)ncc1F 28036,C1(CC#C)(C(=O)NCc2ccc(Cl)cn2)CCN(C(=O)CCSC)C1 28037,c1(C(C)=O)cccc(C(=O)NCC(F)CNC(C2(c3ccc(F)cc3)CC2)=O)c1 28038,c1(SC)nc2ncnc(NCC3(F)CCN(C(=O)C(C)C4CCCO4)CC3)c2s1 28039,C1(CNC(C2C(OCC)C2)=O)CC(C(C)C)CCN1C(=O)CCS(=O)(=O)CC 28040,c1(OC)ccc(OC)c(C=CC(=O)N(C(C)CNC(c2cc(OC)n[nH]2)=O)C)c1 28041,Cc1ccc(C(=O)NC2CCOCC2NC(=O)CCc2ccoc2)cc1N 28042,C1(C(=O)NC(CCOC)C(C)C)CCCCC1(C)NC(c1c[nH]c(=N)c(C)c1)=O 28043,c1(C(N2CCC(NC(CC)=O)C2)=O)ccc2c(c1)CN(C1CCC(=O)NC1=O)C2=O 28044,N1(C(C)=O)CCN(C(C2CC(N(C)C)CN2C(=O)CC2CCCC(=O)N2)=O)CC1 28045,C1(C(N(CC(C)CNC(=O)CC2CCCSC2)C)=O)CC2COCC2C1 28046,CCCS(=O)(=O)C(C)C(=O)N(C(C)CCNC(c1cc2sccc2n1C)=O)C 28047,N(C1CCc2c(Br)cccc21)c1cc(NC(C(n2ncc(C)c2)C)C)ncn1 28048,c1(NC(=O)NC(CC)C)ccc(NCC(F)(F)C(C)C)c(C)c1 28049,c1(C(=O)NC(CN(C(CC(=C)C)=O)CC)CC)cc(OC)c(OC(C)C)c(Cl)c1 28050,c1(C(c2nnnn2CC(F)F)NCCC(C)CO)ccc(Cl)c(F)c1 28051,N1(C(c2c(CC)sc(=N)[nH]2)=O)CCCOC(CCNC(=O)C(C)CC2CC2)C1 28052,CN1C(C(c2nnnn2C2CCCCC2)NC2CCCSCC2)CCS1(=O)=O 28053,c1(OCC(N2C(CNC(=O)C3=COCC3)CCC2)=O)ccc(F)cc1Cl 28054,N1(C(CN(C)Cc2ccccc2)=O)CC(CNC(c2cc[nH]n2)=O)C(O)C1 28055,CN1c2ccc(C(=O)NCCCNC(c3coc(Cl)c3)=O)cc2C(C)(C)S1(=O)=O 28056,C1(NC(c2c(CC)non2)=O)CCN(C(C2COCC(C)O2)=O)C1C1CC1 28057,N1(C(C(N)=O)=O)CC2(CCC2CNC(C2CCCS2)=O)C1 28058,c1(CC(C(=O)OC)NCc2ncc(C)cn2)ccc(OC)cc1Cl 28059,c1(C(N(CC(C)NC(C2(c3ccoc3)CC2)=O)CC)=O)cc(C)cc(C#N)c1.C 28060,CN=c1[nH]cc(C(=O)N(C2CCN(C(c3ccncn3)=O)C2)C)s1 28061,c1(C(=O)NCC(CN(C(C2(C(=O)NC)CC2)=O)C)(C)C)[nH]c(C)c([N+](=O)[O-])c1C 28062,N1(C(CC2(C=C)CCCCC2)=O)CC2(C1)CN(C(=O)C(C)NC(=O)NC)CCO2 28063,c1(CCCC)ccc(CC(=O)NC(CNC(=O)CCCCOCC)C2CC2)cc1 28064,c1(C(C)NC(C2C(C#N)CCC23CCC3)=O)ccc2nc(O)[nH]c2c1 28065,C(=O)(CC1=CCN(C)CC1)NCC(C#C)OC.O1NC(=O)C2CC2C1C 28066,c1(C(N2CCN(C(CSCCCC)=O)CC2C(C)C)=O)cccc2cncn12 28067,CC1CCCCC1C(=O)N(C1CCCCC1)CCNC(=O)COc1ccccc1 28068,N1(C(c2nc(OC)oc2)=O)CCC2(CCN(C(=O)Cn3cc(CO)nn3)C2)C1 28069,C1(CNC(c2c(CCC)n(C3CCCC3)nc2)=O)CC2(CC2)CN1C(=O)COC 28070,N1(C(c2c(O)ccc(C#N)c2)=O)CCC2(CCCC2NC(=O)CC(F)(F)F)CC1 28071,c1(CC)cc(C(c2nnnn2CN2CCOCC2)NCCCc2cccs2)on1 28072,c1(OC)ccc(C)nc1C(N1CC(OC)C(NC(=O)COc2ccsc2Cl)C1)=O 28073,C(=O)(C(C(C)(C)C)n1ccnn1)N(CC(CC)NC(c1csc(=NC)[nH]1)=O)C 28074,Cc1[nH]nc2c1CCC(C(=O)NC1CCCN(S(=O)(=O)c3ccc(Br)cc3)C1)C2 28075,C1(O)(C(C)NC(COC)=O)CCN(C(=O)Cc2ccccc2CC#N)C1 28076,c1(OC)ccccc1NC(N1CCN(c2cc(SC)ncn2)CC1)=O 28077,C1(NC(=O)CC2CC3(CC3)C2)CC(CNC(c2csc(Br)c2)=O)C12CCC2 28078,c1(C(=O)NC2CC(NC(c3n(C)ccc3)=O)C23CCC3)cc(N=S(C)(C)=O)ccn1 28079,N1(S(CC(=O)OC)(=O)=O)CCCC2C1CCN2Cc1ccc2occc2c1 28080,C1(OC)CN(C(=O)Cc2nccn2C)CC1NC(C1CCOCC1)=O 28081,CCCCS(=O)(=O)C(=O)NC(CNC(=O)C(=Cc1cccnc1)F)CC 28082,C(=O)(CC1=CCCCC1)N1CC(NC(c2cc(N)c(Cl)nc2)=O)C(C(F)(F)F)C1 28083,c1(OC)ccc(C(=O)NCC2CC(O)CN2C(=O)C(F)=CCCF)nc1OC 28084,S(=O)(=O)(c1[nH]c(=NCCCCCN(C)C)ccc1Br)N1C(C)c2cccnc2CC1 28085,Cc1cn2ccc(C(=O)NCC3CCCC3NC(c3sccc3C)=O)cc2n1 28086,N1(C(C(C)(C)NS(C)(=O)=O)=O)CCOCC(NC(c2coc(Br)c2)=O)C1 28087,Cc1ccc(NC(c2nnnn2C(C)C)CC2CCCOC2)cc1C 28088,C=CC1CN(C(=O)CCN(C(=O)CCCCCC)CC)CCO1 28089,CCC(C)(C)CCCC(=O)N1CC(NC(=O)COc2ccccc2)CC1(C)CC 28090,Cc1cc(Br)oc1C(=O)NCC1COC(CNC(=O)C=Cc2cocn2)C1 28091,C1(CC)CCCCCN1C(=O)Cn1cc(CO)nn1.c12cc(ccn1)NC2=O 28092,c1(C(=O)NCC(CNC(c2c(N)nc(Cl)cc2)=O)CO)ccc2nonc2c1 28093,CCC(C)C(O)C(C)C(=O)N(C)CC1CCCN1C(C12CCCN(CC1)C2)=O 28094,C1(C(N(C)CC2CN(C(c3cn(C4CC4)nn3)=O)CCO2)=O)CCC=CCCC1 28095,C1(CCC(=O)NCC(CC)(C)NC(c2cc(Cl)ccn2)=O)NC(=O)NC1=O 28096,CC1CN(C(=O)C2=CCSC2)CC2(CCN(c3nnc(C(N)=O)s3)C2)O1 28097,C(CN=c1nn[nH]n1-c1ccccc1)N(C1CC2CC2C1)CC 28098,C1(C(=O)NCC2CCN(C(CCC(C)C)=O)CC2)COC(C)(C)CO1 28099,N1(C(CCC(CC)CC)=O)CC(C2CCCCN(C(C3CCSC3)=O)C2)C1 28100,c1(C(N(CCNC(c2cscc2Br)=O)CC2CC2)=O)cc2ncccc2[nH]1 28101,C12(C(=O)NC3C(NC(C(C)OCC(F)(F)F)=O)COC3)CC3CC(C(=O)N1)C2C3 28102,C12(CNC(c3[nH]c(CC)c(Cl)n3)=O)CCC(C1)N(C(c1ccc(OC)nn1)=O)C2 28103,C1(NC(c2c(NC(C)=O)cccc2)=O)CCN(Cc2ccc(O)c(O)c2)CC1F 28104,N1(C(c2c(CNC(=O)N(C)C3CC3)noc2)=O)CCC(C(=O)OC)C(C)C1 28105,C12(C(N(C(CN(C(CNC(CCC)=O)=O)C)C)C)=O)CC1COC2(C)C 28106,C1(C(C)=O)CCC(F)(F)C1O.N12CCN(CC1C)CCN(C(C)(C)C)C2=O 28107,C1(CN(CC=C)C)CCCN(C(C2CCCCN2C(c2ccnc(F)c2)=O)=O)C1 28108,C(C(C)(C(=O)Nc1conc1C)NC(c1ccc(C#N)o1)=O)SC 28109,C(C[Si](C)(C)C)NC(CN(CC#C)C(c1cc(Cl)cs1)=O)=O 28110,C(CC(N)=O)(C(=O)N1CC(C(=O)NC2CC2)C1)NC(c1nccc(CC)c1)=O 28111,c1(C(=O)NCC2CN(C(CCSCC)=O)CC2O)cc(CC)cnc1O 28112,C1(NC(CCOCCOCC)=O)CN(C(=O)C(C)CF)CC1F 28113,N1(C(CCC(=O)N(C)C)=O)CCC(C2CCN(C(c3ccc(F)cc3Cl)=O)C2)C1 28114,c1(CCC(=O)NC2C(NC(Cc3c(C)scc3)=O)COC2)cccc(N(C)C)c1 28115,c1(C(N(c2n(CC)nc(C)c2)C2CC3CNC2C3)=O)cc(F)ncc1NC(C)=O 28116,N1(C(CC)=O)CCC(C(=O)NCC(CC)NC(=O)CC(O)c2ccccc2)C1 28117,c1(-n2cc(C(C(OC)OC)C)nn2)ccc2ncc(Br)cc2c1 28118,N1(C(C(C2CC(F)(F)C2)OC)=O)CCC(NC(c2ccns2)=O)CC1C 28119,N1(C(c2cc(CC)sn2)=O)CCN(C(c2c[nH]c(=NC)s2)=O)C(C2CCCC2)C1 28120,C1(C(=O)NCC(C)CN(C)C)C2CCCC2CN1C(C1CC=CC1)=O 28121,CCCCCCC(C)(c1nnnn1C(C)(C)CC)NCC=C1CCSCC1 28122,C=CC(C)(O)CC(=O)N(C1CCCCN(C(c2nc(OC)cc(OC)n2)=O)C1)CC 28123,c1(NC2C3CN(C(C4N(CCC)CCCC4)=O)CC32)nnc(C)c(C)n1 28124,C=C(C)C(C)(C)C(=O)NCC(C)(O)CNC(c1ccnc(C(C)(C)C)c1)=O 28125,N1(C(c2cccc(C)c2F)=O)CCC2(C1)CN(C(=O)C=Cc1cc[nH]c1)CCO2 28126,c1(CN=C(NCC2(C)CC2)NC2CCS(=O)(=O)C2)ccc2c(c1)OCCCO2 28127,N1(C(CCCCCNC(Cc2c(C)n(C)cn2)=O)=O)Cc2cccc(F)c2C1 28128,N1(C(CSCC2CCCO2)=O)CC2CCCC(C(=O)NCc3[nH]c(=N)sc3)C2C1 28129,N1(C(C=C(C)C(F)F)=O)CCC(F)(C(N2CCCC2C2(C)CC2)=O)CC1 28130,C#CCCCC(C(=O)Nc1ccc2c(c1)OCO2)N(C1CCCCC1C)C 28131,c1(-c2nc(C(C)C)nn2C2CCS(=O)(=O)CC2)ccnc2c(I)cnn12 28132,Cc1c(C(=O)NCC2CCN(C(=O)C(F)=C3CCC3)C2)cnn1CCO 28133,c1(OC)c(C(N2CC(C3CCCN(CCN(C)CCO)C3)C2)=O)cccc1Cl 28134,CC1CN(C(c2cnn3c2SCC3)=O)CC(C)N(C(c2cncs2)=O)C1 28135,C(=O)(C(F)C(C)CNC(c1ccc(C)o1)=O)N(C(CC)C(=O)OC)C 28136,N1(C(C2CCC2)=O)CCC2(CC1)CN(C(c1c(F)cncc1F)=O)CCC2O 28137,c1(C(=O)NC(C(C(C)C)NC(Cc2c(C)ocn2)=O)C)ccsc1S(C)(=O)=O 28138,N1(c2ccnc(N(CCS(N)(=O)=O)C)n2)Cc2cnc(C(F)(F)F)nc2C1 28139,Cc1ccc(N)c(C)c1C(=O)N(CC(O)CN(C(=O)CC(C)C1CC1)C)C 28140,CCC(CC(=O)N(CC(C)C(=O)NC(C)CC1CC1)C)CC(C)C 28141,C1(NC(C=C2CCN(C(C3(COC)COC3)=O)CC2)=O)CC(=O)N(C)C1=O 28142,C1(CNC(C(CCCC)C)(C)c2nnnn2CC(F)F)Cc2ccccc2CO1 28143,c1(C(=O)NC(c2cc(F)cc(Cl)c2)CNC(C2CC(O)C2)=O)n[nH]cc1[N+](=O)[O-] 28144,N1(C(CCCn2c(C)ncc2)=O)CC(NC(=O)CC2COCCO2)CC(C)(C)C1 28145,CON1CC(C(=O)NCC(C(=O)NC(C2(CO)CC2)C)N(C)C)CC1=O 28146,C(=O)(C1=CC2C=CC1C2)N1CCCC(C(=O)Nc2c(C(C)C)nccc2)CC1 28147,C12(CNC(CC=CC=C)=O)CCCCC1CN(C(c1ccc(CO)c(Cl)c1)=O)C2 28148,C(CCN(C)C)(C(=O)NCC1(O)CCOC1)NC(Cn1ncc(CC)c1)=O 28149,C#Cc1cccc(CNC(C2(CCNC(=O)C(c3cnccn3)C)CCC2)=O)c1 28150,N1(C(C2(C)CCCOC2)=O)CC2CCN(C(c3ccc(Cl)cc3O)=O)C(C2)C1 28151,CC1(C)CC1(C#N)C(N1CC2C(NC(=O)Cc3cn[nH]c3)C2C1)=O 28152,c1(C(=O)NCC2C(C)CN(C(c3nnc(C(C)(C)C)s3)=O)C2)cc(C#N)cn1C 28153,c1(C(=O)NC2C(C)(C)CCN(C(C3(C)COC3)=O)C2)cc2nn[nH]c2cc1F 28154,C(=O)(C1=CCCC(C)(C)C1)N(C1CCN(C(C2(S(C)(=O)=O)CCCC2)=O)C1)C 28155,CC(C)(C)C(CNC(C1CCC(F)(F)C1)=O)NC(c1cnc(-c2ccco2)s1)=O 28156,N1(C(c2cnn(CC)n2)=O)CCCC(C2CCCCN2C(=O)CNS(C)(=O)=O)C1 28157,c1(C(=O)OC)ccc(NC(=O)CC2CC(NCc3ccc(O)cn3)C2)cn1 28158,CN(S(=O)(=O)N1CC(O)CO1)CC1COCCC1(F)F 28159,Cc1csc(C(=O)N(C(C(=O)NCC2(S(C)=O)CC2)C2CC2)C)c1 28160,C12(C(=O)NCCNC(c3cccc(CC4CC4)c3)=O)CCC(F)(CO1)C2 28161,C(=O)(C(O)CCn1cncn1)NC(C(C)NC(c1cnn(CC2CC2)c1)=O)(C)C 28162,C1(OC)(CNC(=O)C=Cc2cccs2)CCN(C(C2C3CCCCC23)=O)C1 28163,N1(C(C2C(c3ccn(C)n3)C2)=O)CCC2(NC(=O)CCc3cccnc3)CC2C1 28164,C(=O)(CS(=O)(=O)CC(F)(F)F)NC1(COC)CCN(C(C(CC)(C)O)=O)C1 28165,c1(C(N(CC(C)NC(C2CCCO2)=O)C)=O)ccc(N)c(C(F)(F)F)c1 28166,C1(C(=O)NC(C(C)C)(C)CNC(=O)C(C)(C)N(C)C)CCCC(=O)N1C 28167,n1(CCC)ccc(C(=O)NC2(c3ccccc3)CC(NC(=O)C=C(Cl)Cl)C2)n1 28168,c1(CC)ccc(C(=O)NCC(C)CN(C)C(c2cccn2C(C)C)=O)cc1Cl 28169,c1(C(=O)NCC2CCN(C(Cc3nc(C)sc3)=O)C2)ccc2c(n1)CCC(C)C2 28170,Cn1ncc2ccnc(C(=O)NCC=CCNC(=O)C(O)P(C)(C)=O)c12 28171,c1(NC(C2N(Cc3c(C)c(O)ccc3)CC3(CC3)C2)=O)cnn2ccc(Cl)nc12 28172,Cc1nc(O)sc1C(=O)NC(C)(CSC)C(=O)NC1CCN(C(N)=O)CC1 28173,N1(C(C(=O)N(C)C)=O)CCCC2(CNC(c3sccc3Br)=O)CCCC12 28174,CC(C)C(C(=O)NCC1CN(C(=O)Cc2ccccc2F)CC(C)(C)O1)C(C)C 28175,C(=O)(C(CCSC)NC(=O)C(C)NC(=O)CC)NC(CC=C)C1CC1 28176,C1(NC(c2cscc2Br)=O)CN(C(=O)CCc2cncnc2)CC1(F)F 28177,c1(CNC(c2cc(N3CC(CC=C)(C(=O)OC)C3)ncn2)=O)ccccc1CC 28178,c1(NCC(C)N(C(c2c(COC)cco2)=O)C)ncc(Cl)c(C)c1C#N 28179,c1(C(N2C3(CN(C(C4CN(CCC)C(=O)C4)=O)C3)CC2)=O)cc(F)cc(F)c1F 28180,N1(C(C(=O)NCC)=O)CCC2(CC1)CC2CNC(c1cnc(C)n1C)=O 28181,c1(C(N2CC(C)C(NC(c3cscc3S(C)(=O)=O)=O)C2)=O)ccn2ccnc2c1 28182,C(c1csc2ccccc12)=CC(=O)NC1CCCCN(CC)C1=O 28183,c1(C(=O)NCCCN(C(C2CC(C)C2(C)C)=O)C2CC2)cccc2ncnn12 28184,CC(C)CCCCCC(=O)NC(C1(CNC(=O)Cn2cc(C(F)F)cn2)CC1)C 28185,c1(CC(=O)NCC(C)NC(c2c[nH]nc2-c2ccccc2)=O)cc(F)cc(F)c1 28186,c1(CNC(N2CC(c3ccn(C)n3)OCC2)=O)ccc(I)c(Br)c1 28187,C1(OC)CC(CNC(=O)C(=O)NC(C)Cc2cccnc2)C1(C)C 28188,C1(CC(=O)NC)CN(C(=O)C(O)CC(F)F)CCN1C(c1nc(C)sc1C)=O 28189,N1(C(C(CC2CCCC2)NC(c2c(C)nc(O)s2)=O)=O)Cc2n[nH]cc2C1CO 28190,C1(C(=O)NC2C(NC(C(C)(C)OCC)=O)CCC2)CC(c2cccnc2)=NO1 28191,N1(C(Cc2cc(C)sc2C)=O)CCC2CN(C(C3CC3c3cccs3)=O)C2C1 28192,Cc1c(C(N2CCC(CCNC(C3CC(=O)N(CC4CC4)C3)=O)C2)=O)ncn1C 28193,N1(C(CS(N)(=O)=O)=O)CCOCC(NC(=O)C(F)Cc2ccccc2)C1 28194,Cc1nc(Cl)ccc1CC(=O)N(CC(O)CN(C)C(c1ccn(C)c1)=O)C 28195,Cc1ccc(CNC(N2CCC(NC(C34CC(CO3)C4)=O)C2)=O)cc1 28196,c1(OC)ccc(C(N2CC(O)CC2C(=O)NCc2ccc(Br)c(Br)c2)=O)cc1I 28197,C1(C(=O)NC(CNC(CC2(C)CCCCC2)=O)C2CC2)CCOC(=O)CC1 28198,c1(C(N(CCNC(Cc2cnc(C)[nH]2)=O)CC2CC2)=O)ccc(OC(F)F)nc1 28199,C12(CC(N3CCC(n4cnnn4)C3)=O)CCC1CN(C(C1CS(=O)C1)=O)C2 28200,C1(N(C)C(C2(C)CC2)=O)CCCN(C(C2(C)CCC(=O)N2)=O)CC1 28201,C1(CCC(N2CC(CNS(C)(=O)=O)C2)=O)CCCCO1.C1(=O)CO1 28202,c1(CNC(NCc2cn(C)nc2)=NCCN2CCCC2)ccc2oc(O)nc2c1 28203,N1(C(c2c(C)cncc2C)=O)CCC2C(CCCN2C(=O)C(F)CC(C)C)C1 28204,c1(C(=O)Nc2cnc(C(C)C)nc2)ccc(Cl)c(O)c1 28205,C1(NC(C2CC(=O)NCC2)=O)C2CC(O)C1N(C(=O)C=C1CCC1)C2 28206,CC1CCCCC1(CNC(=O)Cc1sc(O)nc1O)NC(=O)CC1CCCCC1C 28207,N1(C(c2nc(OCC)sn2)=O)CCC(C2(NC(c3cc(CO)[nH]n3)=O)CC2)CC1 28208,CCCCCS(=O)(=O)CC(=O)NC1CCN(C(c2cc(OC)cnc2F)=O)CC1 28209,C1(NC(c2c(OC)n[nH]c2)=O)CC(C)N(C(=O)Cc2nn(C)cc2Br)C1 28210,N1(C(C2(CNC(=O)C(C)S(N)(=O)=O)CC(=C)C2)=O)CCC(C2(C)CC2)C1 28211,c1(C(N(CC(C)O)CCNC(c2cncc(C=C)c2)=O)=O)cnc2scc(C)n12 28212,S(=O)(=O)(c1c[nH]ccc1=NCC1(S(=O)(=O)CC)CC1)NC(CCCC)(C)C 28213,N1(C(c2cncc(OC(C)C)c2)=O)CCC(CNC(=O)C(C)(O)C2CC2)C1(C)C 28214,c1(C(N2CCC3(C(NC(=O)CCBr)C3)CC2)=O)cnc2cc(Cl)ccc2c1 28215,c1(CC(N2CC(OC)C(NC(=O)C(C)S(N)(=O)=O)C2)=O)ccc2c(c1)NC(=O)C2 28216,N1(C(C(CC)SC)=O)CCC2(CC1)CCN(C(=O)C=C(C)c1ccco1)CC2C 28217,CC1=C(C(=O)NC23CCN(C(=O)CC(C)(C)C)CC2C3)CCC1 28218,N1(C(C=CCCC)=O)CCC(CNC(=O)Cn2ccnc2)C(C)C1 28219,C(=O)(CC1OCCc2ccsc21)N1CC(NC(C(CC(C)C)(F)F)=O)CC1(C)C 28220,c1(C(=O)NCC(C2CC2)NC(C(N2CC(C)C2)C)=O)cc2cc[nH]c2cn1 28221,C(=O)(CCCCCN(C(C1CCC1C)=O)C1CC1)N(CC(F)F)CC 28222,C(C)(C)(CC(F)C(=O)NCCc1cccnc1)NC(c1scc(C)c1)=O 28223,c1(C(N2CCCC(NC(C(C)n3cccc3)=O)C2)=O)ccc2c(c1)COC2 28224,C(CC(=O)N1CC(CC(C)(C)C)C1)N(C(=O)C=CC(F)(F)F)CC 28225,C(C(C)(C(C)C)NC(=O)Cc1csc(S(C)(=O)=O)n1)NC(COCCCC)=O.N 28226,C1(NC(C(C#C)(C)C)=O)CCC(C)(CNC(c2coc(C(F)F)n2)=O)CC1 28227,c1(C(=O)NCC2(NC(c3cnn[nH]3)=O)CCOC2)cccnc1SC(F)F 28228,CC1CCC(C)(NC(c2conc2CNC(C2C3CCC(=O)C23)=O)=O)C1 28229,c1(CC(N2CCC2CNC(C2CCC(F)CC2)=O)=O)ccc2c(c1)CCO2 28230,C1(C(N2CC(c3nccn3C)(OC)C2)=O)(Oc2ccccc2)CCS(=O)(=O)C1 28231,C1(NC(C(C)NC=O)=O)CCN(C(c2ccnn2CCF)=O)CC1(C)C 28232,CC1CCCCC1C(=O)NC(C)(C)C=CC(=O)NCC(F)Cl 28233,c1(C(N)=O)ccc(CC(N2CCOCC2CNC(=O)CCC2CCCO2)=O)cc1 28234,C1(CNC(=O)C=Cc2cocn2)CCCC2(CN(C(=O)C(Cl)=CCl)C2)O1 28235,Cc1c(C(=O)NCC2CN(C(=O)C(F)C3CCC3)CCCO2)nn(C)c1N 28236,Cc1cccc2c(C(N3CCC4(NC(=O)CCOC(C)C)CCCC34)=O)coc12 28237,N1(C(C2CCOC2C(=O)NC2(c3nc[nH]n3)CCC2)=O)CCCC1(C)C(=O)N.CO 28238,N1(C(C(C(C)C)SC)=O)CCN(C(=O)Cn2ccccc2=O)CC12CC2 28239,Cc1cccc(C(=O)NCC(F)CNC(c2cnc(CC(C)C)[nH]2)=O)c1C 28240,c1(C(=O)NCC2CCOC2)cc2c(s1)CCN(C(c1cc(Cl)c(Br)cc1Cl)=O)C2 28241,C(=O)(C(F)(F)C(F)(F)F)NC1C(CNC(c2cc(C)n(CCO)n2)=O)COC1 28242,c1(C(=O)NCC)ccc(NC(=O)Cn2cc(CCCNC(N)=O)nn2)cc1C 28243,CC1(C)CC(CNC(=O)CCCNC(N)=O)CN(C(C2(F)CC2)=O)C1 28244,N1(C(C=C(C)C(C)(C)C)=O)CC2CCCCC2(CNC(=O)Cc2ccsn2)C1 28245,C#Cc1ccc(C(=O)NC2CCN(C(=O)CC(C)C(F)(F)F)C23CC3)cc1C 28246,CP(C)(=O)C(O)C(=O)NCCOCCOCCCNC(c1cncc(Cl)c1)=O 28247,C#CC1CN(C(C2CCC2C#N)=O)CCN1C(c1cnc2[nH]nnc2c1)=O 28248,C(=O)(CCCCCCNC(=O)C(C)(CO)NC(C)=O)NC(C(C)NC(C)=O)CO 28249,N1(C(C(F)=CC)=O)CC(COC)CCC1=O.C1(C(N2CCC2C(=O)OC)=O)CCC1C 28250,c1(OC)ccc(CCC(=O)NCCCCNC(c2cccc(CO)c2)=O)c(C)c1 28251,C#CCC(C)(C(=O)NCC(C)S(N)(=O)=O)NC(c1cccnc1NC)=O 28252,Cc1c(F)ccc(CN2CCC(F)(C(=O)NC(c3cccnc3)C)C2)c1Cl 28253,CCCC(CCC)C(=O)NCCN(C1CCCCC1)C(C1CC1COC)=O 28254,c1(C(=O)NCC(CO)NC(c2cc(SC)oc2)=O)ccc([N+](=O)[O-])s1 28255,n1(CCC(N2CCC(C(C)NC(c3ccc(CC)[nH]3)=O)C2)=O)ccc(O)nc1=O 28256,CCCC(C(=O)OC)C(=O)N1CCC(C)(C)C1C(=O)NCc1cnc(O)nc1O 28257,C1(Cl)(C(N(C(C)CNC(=O)COC)CC)=O)CC1.C1CCC1 28258,C(=O)(CCN(OC)C(=O)C(C1CC1)NC(C1(c2ccccc2)CC1)=O)OC 28259,c1(N2CC(C)(C(N(CC(F)(F)F)C)=O)C2)ncnc2sc(-c3ccccc3)nc12 28260,C(=O)(C1=NOC(C)(C)C1)N1CC(C(=O)NCC(COC)C(C)C)C(F)C1 28261,N1(C(c2cnn(C3COC3)c2)=O)CCN(C(c2csnc2Br)=O)CC1 28262,c1(C(=O)OC)cc(CCNC(=O)C(F)C2CC(NC(c3ccc[nH]3)=O)C2)on1 28263,C(=O)(C(C)(C)C(F)F)N1CCCC(CCNC(C2C(C)(C)C2(F)F)=O)C1 28264,N1(C(COCCC)=O)CCCC12CCN(C(C1CCC(C)=C(C)C1)=O)C2 28265,N1(C(c2c(CC)ncs2)=O)CCCC(C(C)NC(c2c(C)nnn2C)=O)C1 28266,C(CCCCCNC(=O)C(Br)=C(C)C)N(C(c1c(CC)cco1)=O)C 28267,c1(C(=O)NCC#CCNC(=O)C=CC2CCCO2)cc2ccccn2n1 28268,c1(C(=O)NC(CC(C)NC(=O)Cn2cc(Cl)cn2)C)ccc2c(c1)CCC2(F)F 28269,S(=O)(=O)(c1ccc2c(c1)COCC2)N1CC2C(C)(C)C2C1 28270,C1(C(=O)NC2CCCC(NC(=O)CSCC(F)(F)F)C2)(CC)CCC(O)CC1 28271,c1(NC(C2C(C(=O)NC(COC)CO)C2)=O)cnn2c(-c3ccccc3)ccnc12 28272,C[Si](C)(C)c1ccc(-c2ccc(Cl)c(S(N)(=O)=O)c2)cc1 28273,Cc1ccccc1CC(C)C(=O)NCCC1(NC(=O)CCSCC(N)=O)CC1 28274,CS(=O)(=NC(=O)CC1CCCCS1(=O)=O)c1ccccc1 28275,c1(C(=O)N)c[nH]cc(F)c1=O.N1(C(C2C(C)C2)=O)CCCC(n2cc(C)nn2)C1 28276,C12(NC(CC(CC)C(C)C)=O)CCCC(CN(C(c3cccn3C)=O)C1)C2 28277,N1(C(CCC(C)(C)F)=O)CC2CCC(C1)N2C(C1(C)CSC1)=O 28278,c1(OCC(=O)NC)cccc(CO)c1.C1CCN(C)C(=O)O1 28279,Cc1nnc2n1CCN(C(=O)NCc1ccc(C3CCC3)nc1)C2 28280,N1(C(C2CC(C(C)C)OCC2)=O)C2CCCC1CN(C(c1cccc(O)n1)=O)C2 28281,C1(NC(C(C)(C)O)=O)CC2CC(NC(C3CCCN(CC(F)(F)F)C3)=O)C1C2 28282,C(=O)(C(CCCOC)NC(=O)CSCCOC)N1C(CC)CC1 28283,CCC(CCCC(=O)NC1(CC)CCCC1)NC(C1(NC(N)=O)CC1)=O 28284,N1(C(CC(CNC(C2(C(C)C)COC2)=O)CC2CC2)=O)CC2CC(OC)CC1C2 28285,CCC(CC(=O)N1CCC(C(C)O)CC1)NC(=O)C(=CC1CCCC1)C 28286,NS(=O)(=O)CCC(=O)N1CC(Cn2cc(C3(O)CCOC3)nn2)C1 28287,Cc1nc(C(F)(F)F)ccc1CNC(=O)C=CC(C)NC(C1CC1(C)C)=O 28288,N1(C(C2(CCOC)CC2)=O)CCC2C(C1)CN2C(=O)CC1(C(F)(F)F)CC1 28289,C#CC1CN(C(=O)CC(CC)N(C(=O)C(C)CC(C)C)C)CCN1C 28290,N1(C(CCN(C(C2=CC(C)(CC)C2)=O)C(C)C)=O)CCCC(C)(OC)CC1 28291,Cc1ccc(CN2C(C(=O)NCC3CCC(O)CC3)CC3CC23)c(Cl)c1Cl 28292,C1(C(=O)NCc2ccc(CNC(C3C(C)N(C)CC3)=O)cc2)CC2CCC1CC2 28293,N(C1CC(C)n2ccnc21)C(CCC(Cn1cc(CNC(CC)=O)nn1)(F)F)=O 28294,C1(C(=O)NCC(C=C)O)CCN(C(C2CN(C)CCO2)=O)CC1(C)C 28295,C(=O)(C1COc2ccccc21)N1CC2(C(NC(C=CC=CCC)=O)CC2)C1 28296,C1(C(=O)NCC(N2CCN(C(c3ncccc3F)=O)CC2)C)CC2(CCC2)C1 28297,C1(CNC(C2(CC#C)CCCC2)=O)CCCN(C(=O)C(C)(C)O)C1 28298,N1(C(CNC(CNC(c2cc(C)sc2N)=O)=O)=O)CC2CCCCC2C1C 28299,C(=O)(C(C)(C)C(F)(F)F)NCCC1CCC(NC(CCC(=O)NCC)=O)C1 28300,CCCCCCCC(=O)N1CC(CNC(=O)C(c2ccc(Cl)cc2Cl)O)C(C)C1 28301,C1(N(C)C)CCCCC1C(=O)NC1CC(C)(NC(=O)CCC2CC2(C)C)C1 28302,C1(NC(CCCCN(C(C)C)C)=O)CC2C1CCN2C(C1CCNC1=O)=O 28303,N1(C(CCCOCC=C)=O)CCC2(CCCN(Cc3ccc(Cl)c(F)c3)C2)C1 28304,N1(C(C(CC)C#N)=O)CCCC(C(=O)NC2COCC2CO)CC1 28305,N1(c2nnc(CC(C)C)n2CC(C)C(F)(F)F)CC2C3CCC(CC3)C2C1 28306,Cc1ccccc1CC(N1CCCC(CCNC(c2cncn2C(C)C)=O)C1)=O 28307,c1(OCC#C)cncc(CN2CCC(SC)CC2)n1 28308,C(CC(C(=O)NCCC1C=CCC1)NC(=O)CC1(O)CCOCC1)N(C)C 28309,c1(C(=O)NC2(CC=C)CCN(C(=O)CSCCC(C)C)C2)cnc(C)c(C)c1 28310,CC1C2CCC(C2)C1C(N1CCC(C)(CC(N2CCC2C2CCCC2)=O)C1)=O 28311,N1(C(C=C(CC)C)=O)CCC2CCC12CNC(=O)Cn1cc(Br)ccc1=O 28312,c1(-n2c(C3CCC(C(C)OC)CC3)nc(CCCCCC)n2)cc(C)ccc1C 28313,c1(C(=O)NCC(CC=C)NC(C2CC(F)C2)=O)ccc(C(F)(F)F)cn1 28314,c1(C(=O)OC)cncc(C(=O)NC23CC(NC(C4CCCNC4=O)=O)(C2)C3)c1 28315,C(C(C(=O)NCc1nc(C2CC2)n[nH]1)C(C)C)NC(C(C)SCC)=O 28316,C(C(CC1CCCC1)C(=O)NC1CCC(C)CC1)NC(COC(C)=O)=O 28317,CC(C)(C)COCC(=O)NC(C(=O)NCCOC(F)(F)F)C1(C)CC1 28318,N1(C(C2C(COC)CC2)=O)CCN(C(c2ccccc2Cl)=O)CC(O)C1 28319,CCC(C(=O)OC)C(=O)NC1(CNC(c2cccc(SC(F)(F)F)c2)=O)CCC1 28320,C1(NC(CC=CC(C)(C)C)=O)C2CCC(F)(F)C12.C12CCC(CC1)C(=O)NOC2 28321,c1(-c2nc(CN(C)C)nn2C2CC2)cc(F)c(Cc2cccc(O)c2F)c(F)c1 28322,N1(Cc2ccc(C#N)cc2)CCOC2(CCCN(C(=O)Cc3cccnc3)C2)C1 28323,C1(NC(C(C)C2CCC2)=O)CN(C(c2cncn(C)c2=O)=O)CC12CC2 28324,C1(NC(CCC(C)c2ccccc2)=O)CC=C(C(=O)N2CC([N+](=O)[O-])C2)C1 28325,C(C(C)C(=O)N(C(C)CC(=O)NCCOCC(C)C)C)OCC 28326,N1(C(CCC2CCC(=O)N2)=O)CCN(C(=O)CSc2ccncc2)C2CCC12 28327,C(=O)(C(F)CC(C)(C)NC(c1ccc(O)cc1)=O)N1CC(C#C)C(O)C1 28328,N1(C(C2C3CN(C(c4cc(OCC)c(Br)cc4)=O)C2C3)=O)CCC(C)C(F)(F)C1 28329,N1(C(c2c(CNC(c3cc(C(C)C)[nH]n3)=O)occ2)=O)CC2(CSC2)C1 28330,N1(C(C(C)CS(C)(=O)=O)=O)CCN(C(C2(C)CCN(C)C2=O)=O)CC(C)(C)C1 28331,CCCCCC(C)(C)C(=O)Nc1cccc(NC(=O)C(C)(CC)CCCC)c1 28332,C1(C(=O)NCCN(C(C=C2CCC(C)C2)=O)C2CC2)(CO)CC(C)(C)C1 28333,C=CCC(CC(F)F)NC(=O)C(CCC1CC1)NC(c1ccncc1CC)=O 28334,C1(C(N2CCC3(C(C(=O)NC4(CC5CCC5)CC4)C3)C2)=O)CC2(CCO1)CC2 28335,C1(NC(C(c2ccc(Cl)cc2)(C)C)=O)CN(C(C2CC(C)(C)C2)=O)CC(F)(F)C1 28336,CCS(=O)CC(=O)NCCN(CCOCCO)C(c1cccnc1OC)=O 28337,n1(CC(=O)NCC2C(CNC(C3CC(CC)C3)=O)C2)ccc2ccccc2c1=O 28338,CC1=C(C(=O)N2CCCCC2C2CCN(C(C3CCOC(=O)N3)=O)CC2)CCO1 28339,O(NC(=O)CN=c1cc(C)c(S(=O)(=O)NC2CCCc3ccoc32)c[nH]1)CC 28340,c1(C(N2C(CN(C)C(C3CC3(C)C)=O)CCC2)=O)ccc(F)c(O)c1F 28341,c1(C(=O)NCCCC(C)NC(C2(CO)CCCO2)=O)cc2cccnc2nc1O 28342,c1(N2CC(C(N)=O)(CNC(=O)CC3CCC(F)(F)C3)C2)ccc2nccnc2n1 28343,C1(C)(C(N2CC=CC(NC(C(CCC)=CCC)=O)C2)=O)CCS(=O)(=O)CC1 28344,C(=O)(C(C)(C)CCC(=O)OC)NCCOCC1CCCN(C(C2CC(=C)C2)=O)C1 28345,C1(C(N(C2CC(C(=O)NC3CCCC3F)C2)C)=O)CCOC1C(F)F 28346,C1(COCC)CCCN(C(=O)C(Cn2cccn2)NC(c2ccc(C#N)o2)=O)C1 28347,C(=O)(Nn1nnc2c1CCCC2)C1C2(CC(NC(C(C)(C)OCC)=O)C2)C1 28348,C(=O)(C1=CC2(CCN(C(=O)CN3CCNC3=O)C2)C1)Nc1cn(CC)c(=O)cc1 28349,c1(N(C(c2cccc(Br)c2)C(=O)NCC(F)F)C)cccc(Br)c1 28350,c1(C(=O)NCCC(CNC(C2COCC2(C)C)=O)OC)cc2nccnc2[nH]1 28351,C(=O)(CS(=O)C(F)(F)F)NCC(C1CCC1)NC(CNC(CC(C)(C)C)=O)=O 28352,C(CCC(C)(C)C(=O)Nn1nnc(C)c1C)NC(C(CC#C)O)=O 28353,N1(C(C2C(C(C)C)OCCC2)=O)CCN(C(=O)C(C)(C)c2ccsc2)CC(O)C1 28354,CCC(C)C(O)C(C)C(=O)N1C2CCC1C(NC(=O)CCNC(C)=O)C2 28355,N1(C(C2C(OCC)C2)=O)CCCC(C)(C)C1CNC(c1cnn(CC)n1)=O 28356,C1(NC(C(CC=CCC)C)=O)C2CCC1CN(C(=O)CC1CC(F)C1)C2 28357,N1(C(C)CSc2cncn2C)CCC(O)(Cn2cc(-c3cncc(F)c3)nn2)C1 28358,c1(CNCC(=C)Cl)csc(C2OCCO2)c1 28359,C1(C(=O)NCCC=CCCC)CCN(C(c2cncc(C#N)c2)=O)C(C)(C)C1 28360,c1(C(N2C(CC)C(NC(c3cccnc3S)=O)CC2)=O)ccc(OC)c(Cl)c1F 28361,CC1(CNC(C2(CF)CCOCC2)=O)COCCN(C(C2CN(C(N)=O)C2)=O)C1 28362,C1(C(=O)NCCC(C)N(C)C(c2ccc(C3CC3)o2)=O)C2CC(F)(F)CC12 28363,Cn1nnc(C(c2nnnn2CC2CC2)NCc2ccnn2C2CC2(F)F)n1 28364,Cc1nc(N2CCCC(NC(c3cc(C)c(F)cc3C)=O)C2)c2c(n1)CCC2 28365,CCC(C(=O)NC1(C)CCN(C(C2CCN2CC)=O)C1)C(C)O 28366,c1(NC(C)=O)ccc(F)c(C(C(=O)CC2(CNCCC)CC2)=O)c1.N(C)(C)CC 28367,N1(CC(=O)N(C2CCN(C(=O)Cn3ncn(C)c3=O)CC2)CC)CCCCCC1 28368,C(=O)(CCC(=O)NC1(CO)CN(C(C2COCC(C)O2)=O)C1)N(CC)CC 28369,C=CCC(C)(C)C(=O)NCC1(O)CC(NC(c2nnn(C)n2)=O)C1 28370,C1(CNC(C2(CC)CC2(F)F)=O)CCCN(C(C2(C(C)(C)C)CCC2)=O)C1 28371,C1(C(=O)NC(C2CCN(C(=O)C(n3cc(Cl)cn3)C)CC2)C)CCCCC(=O)C1 28372,N1(C(C(CCC)(C)O)=O)CC(C)(C)OC2(C1)CN(C(=O)C(C)C(C)COC)C2 28373,N1(C(C=C(CCN(C)C)Cl)=O)CCC2(CCN(C(c3ncccc3N)=O)C2)C1 28374,C1(C(N2CCN(C(c3ccc(C(C)=O)nn3)=O)CC2)=O)CCc2ncncc2C1 28375,c1(N(C)C)ccc(C(N2CC3C(NC(c4nc(Br)c[nH]4)=O)C3C2)=O)nn1 28376,c1(C(=O)NCC2N(C(c3cc(C(C)=O)oc3)=O)CC2)c(Br)ncn1C 28377,C(=O)(C1=NOC(CNC(=O)CC2C=CCC2)C1)N(C(CCO)C(F)F)C 28378,c1(C(=O)NCCC2CC(NC(C=Cc3ccc(C)o3)=O)C2)nccn2cnnc12 28379,C1(C(N2CCN(C(c3cnc(Cl)s3)=O)C3C2C3)=O)CCc2ccccc2CC1 28380,c12ccc(cc1OC)c(=O)[nH]2.c1(SCCCC)cn(C)nc1C(C)(C)C 28381,N1(C(C(C)(C)OC)=O)CCN(C(=O)CC2(c3ccccc3)CCOCC2)CC1 28382,N1(C(C=CCCC)=O)C2CCC1C1CC1(NC(C1CCCC(F)(F)CC1)=O)C2 28383,c1(OC)cc(CN2CCN(CC(=O)Nc3cccc4sccc34)CC2)c(F)cc1F 28384,C(CCC(=O)NCC1CN(C(c2occc2Br)=O)C1)N(C(C)=O)C 28385,Cc1nc(C)c(C(=O)NCCN2CCC(NC(=O)CS(N)(=O)=O)CC2)[nH]1 28386,Cc1ccc2c(C(N3CC(NC(=O)COc4ccccn4)C(C)C3)=O)csc2c1 28387,C1(C(=O)NCC2C(NC(c3nccc(SC)n3)=O)CCC2)CN2CCN1CC2C 28388,Cc1ncn(C)c1C(c1nnnn1Cc1ccco1)NC1CCC(C)(C)C1 28389,N1(C(C(C)=C(C)C)=O)CCN(C(c2cc(C#N)ccc2C)=O)C2CCC12 28390,N1(C(c2c(CCC)n(C)nc2)=O)CCN(C(=O)C(OCC)OCC)C(C)C1 28391,C1(OC)CC2(C1)CC(NC(c1cnn(CCNC(=O)CC3CCC3)c1)=O)C2 28392,C1(N(C)C)(C(=O)NCC2C=CC(NC(c3cccnc3S)=O)C2)CCCCC1 28393,N1(C(c2cn(CCC(C)C)nn2)=O)CCC(NC(=O)CCC(C)(C)O)C(C)C1 28394,N1(C(CNC(C)=O)=O)CCCC(N(C)C(C2COCC(=O)N2C(C)C)=O)CC1 28395,C1(C(=O)NCC2CC(F)CN2C(c2cc(Br)c[nH]2)=O)CCCC12CCC2 28396,c1(COCC)ccc(F)cc1.c12ccc(cc1)OC1CCN(C1)CCCCN2 28397,c1(C(N2CC3C(NC(c4c(CC)nco4)=O)(CC3)C2)=O)cc(N)c(C)cc1Cl 28398,c1(C(N2CC(NC(CN(C)CC)=O)C3(C2)CC3)=O)cc(C)c(C)cc1C 28399,c1(NC(CC)COC)ccc(S(=O)(=O)NCC(N2CCOCC2)C)cc1Br 28400,c1(NC2C(CCC)C2)ncnc(NCc2cc(C(F)F)on2)c1C 28401,C(=O)(CS(=O)(=O)CC1CCCO1)NC1(CNC(C(C)n2cncn2)=O)CCC1 28402,c1(C(=O)NC(C2CCOC2)C#C)oc(CNC(=O)CNC(=O)CC)cc1C 28403,N1(C(C2CCC(C)CC2)=O)CC2CC(C1)N(C(=O)CS(=O)(=O)N(C)C)C2 28404,c1(C(=O)OCC(C2CCC(F)(F)C2)C(=O)OCC)cc2ccsc2n1C 28405,C1(NC(C(C)OCCOC)=O)CCC2(CCN(C(c3coc(C)n3)=O)C2)C1 28406,n1(CC(=O)NC(C2CCCN2C(=O)CC2CCNC2=O)C2CC2)ccsc1=N 28407,CC1CC2(CC(C(=O)NCC(O)C(=O)NC3(CO)CC=CC3)C2)C1 28408,C1(CNC(CCC2(NC(CSC)=O)CCCC2)=O)CCCCC1(C)C 28409,C1(N(C(C(CSC)O)=O)C)CN(C(c2c(O)cccc2F)=O)CC12CC2 28410,C=CC1(C(=O)NC2C(C)C2(C)C)CCN(C(c2cnnc(O)c2)=O)C1 28411,c1(CCC(N2C(C(=O)NC3(CC)CCOC3)CCCC2)=O)ccc(OC)c(F)c1 28412,N1(C(C2CC(NC(C3CC3Br)=O)C2)=O)CC(O)(c2cnn[nH]2)C1 28413,C1(NC(c2cn(CCC)nc2)=O)CCCCCC1NC(=O)C(F)(F)c1cncs1 28414,C(=O)(CC(F)(F)C(F)F)NC1CCCC(CC(=O)NCc2c(C)nc(C)s2)C1 28415,c1(CC(=O)NCCC2CC(NC(c3c(CC)c[nH]n3)=O)C2)cccnc1OC 28416,C(=O)(C(CC(C)C)N(C)C(c1ccc(O)nn1)=O)NC(CC#C)C(N)=O 28417,c1(OC)cc(C=O)oc(=O)c1.N1(O)CC2CC1CN2C(=O)C(F)(F)F 28418,N1(C(c2ccc(C)c(Cl)c2)=O)CCC2(CC1)CC2NC(C1(C)CCSCC1)=O 28419,C1(CNC(C(C(C)C)NC(C)=O)=O)CN(C)CCN1c1cnc(C#N)cn1 28420,C1(C(C)NC(c2cc(Cl)c[nH]2)=O)CCCCN1C(=O)CCc1cccs1 28421,N1(c2cc(C)nc(Cl)n2)CCC(NC(C2CCC3CCCCN23)=O)C(C)(C)C1 28422,CC1COCCC1NC(C1CC12CC(NC(C1(c3cc[nH]n3)CC1)=O)C2)=O 28423,N1(CC(=O)NC(C)(C)C(F)F)CCN(C(C2SCCS2)=O)CC1 28424,c1(CC(=O)NCCCN(C(C=CC(C)C)=O)CCO)cscc1OC(F)F 28425,c1(C(N2CC(C3N(C(C=CC)=O)CCC3)(O)C2)=O)ccc(Br)cc1[N+](=O)[O-] 28426,C1(NC(C(C)NC(C)=O)=O)COCCC1C(=O)NC1CC(C)(C)C1 28427,N1(C(C2C(C)CC2)=O)CCOC(CC(=O)N(C2CCCCC2)CCO)C1 28428,N1(C(C(CC#C)C)=O)CCC2CN(C(C34CC(c5ccccc5)(CO3)C4)=O)CC12 28429,Cc1cc(NC(C2C3CCC(C3)N2C(=O)COc2cnc(Cl)cn2)=O)cc(F)c1 28430,N1(C(CC2C(C)C2)=O)CC2(CO)CC2(C)C1 28431,c1(C(c2nnnn2CCCF)NC(COC)(C)CCO)cnc2cc(Br)ccn12 28432,C(CCCCS(=O)(=O)CCCO)NCC1N(Cc2c(OC)cccc2)CCC1 28433,C1(CC(=O)NCCC(=O)OCC)C2CC(C2)N1C(c1cc(C)oc1C)=O 28434,Cc1cc(C(N2CCCC(C(N3CC(C(C)(C)C)C3)=O)CC2)=O)cc(O)c1 28435,c1(NC(C2(C)CN(Cc3cccc(C=O)c3Br)C2)=O)csc2nccnc12 28436,N1(C(C(C=C)(C)C)=O)CCN(C(=O)CCN2CCC(F)C2)C(CC(=O)NC)C1 28437,c1(C(N(CCCNC(C2CCC(=O)C2)=O)CC2CCCC2)=O)nnc2ccccn12 28438,C1(NC(C2N(C(c3c(C)cc(CC)o3)=O)CCC2)=O)C(=O)NCCC1C 28439,C#CCC(C(=O)NOCC(=O)NCC(c1cn(C)cn1)O)N(C)C 28440,c1(OCCC)ccc(C(=O)NCc2ccc(CO)c(F)c2)cc1C 28441,c1(C2C(C)C2)csc(C(=O)NCCOCCNC(=O)CSc2cn[nH]c2)n1 28442,C1(NC(C(C)NC(CC)=O)=O)CN(C(=O)CN2CCC(O)CC2)CC2(CC2)C1 28443,c1(C(=O)NCCC(C)N(C)C(c2cccnn2)=O)csc2ccc(F)cc12 28444,c1(CNC(C(N2C(C#N)CCC2)c2ccc(CO)cn2)=O)ccc2c(c1)CCC2 28445,C(C1=NOC2CN(C(=O)C#CC3CCOCC3)CC12)NC(c1c(C)scc1)=O 28446,c1(C(=O)NC(CNC(C2CCC(=C)CC2)=O)C(C)C(C)C)ccc2ncnn2c1 28447,C1(C)(NC(CNC(CNC(c2cnc(C(C)C)o2)=O)=O)=O)CCCC1(C)C 28448,CCCCC(C)CCC(=O)NC1COCC1(C)NC(=O)OC(C)(C)C 28449,N1(C(c2cc(C)sc2C)=O)CC(C)OC2(CCN(C(C3CC3C(C)C)=O)CC2)C1 28450,c1(N2CC(C(=C)C)OCC2)nc(=NCCc2ccoc2)[nH]c2c1cnn2C 28451,C(=O)(C1CCCc2c1ncn2C)NCC(C)(CO)NC(c1cc(C)on1)=O 28452,N1(C(c2ccc(SC)o2)=O)CCC(NC(C2CCN2CS(C)(=O)=O)=O)C1C 28453,c1(Cn2cc(C3CC(NC(C4(CC)CCCC4)=O)C3)nn2)cc2n(n1)CCCO2 28454,c1(OC)cc(C(=O)NC2CCC(N(C)C(c3cccc(=O)n3C)=O)C2)c(F)cn1 28455,C1(CC(=O)NCCNC(C)=O)CC2(C1)CN(C(c1cc(C)cs1)=O)C2 28456,C1(NC(C2ON=C(C)C2)=O)CC2(C(=O)NCC3(C4CC4)CCC3)COC1C2 28457,C1(C(N(CCN(C(C)C)C(c2ncc(Cl)n2C)=O)C)=O)CCC2CC2CC1 28458,N1(CC(=O)Nc2cc(C)no2)CCC(C)(CNC(c2ccc(F)cn2)=O)CC1 28459,N1(C(C2CC(CC)N(C(=O)Cc3cn(C)cn3)CC2)=O)CCC(F)(F)C(O)C1 28460,CCCCC(C)(F)C(=O)NCC1(O)CCN(C(=O)CC=Cc2cccc(F)c2)C1 28461,c1(NC(c2n(C)ccc2)=O)ccc(CN2CCSCC2)cc1 28462,C1(CC(N2CCC(NC(c3ccc(C4(C(=O)O)CC4)s3)=O)C2)=O)CCCOCC1 28463,N1(C(c2c(OC)cnnc2)=O)CCC2(CCN(C(=O)C(N=[N+]=[N-])C(C)C)C2)C1 28464,C12(CCS(=O)(=O)CC1)C(=O)N2.c1(CC(C(=O)NCC2CCC2)N)ccc(Cl)cc1Cl 28465,n1(CC)cnc2c(NCCc3cc(F)c(F)c(F)c3)[nH]c(=NC(C)CF)nc12 28466,c1(CC)cc(CNC(=O)C(c2ccc(-c3nn[nH]n3)cc2)O)cc(F)c1 28467,c1(C(N(CC(C)(C)CNC(c2ccc(C(F)F)o2)=O)CC)=O)cnnc(C)c1 28468,C#CCCCCC(C(=O)NC(C)CC)N1CCC2CCC(C1)N2C 28469,C1(NC(c2scc(C)c2)=O)CN(C(c2ncncc2Cl)=O)C2(CCOCC2)C1 28470,C(COC)(CCCC)NC1(C)CN(C(C=CCOC)=O)C1.C1C(=O)N1 28471,C1(CCC)COCCN1C(c1ccn(CCNC(=O)COC2CC2)c1)=O 28472,C(=O)(C1=C(Cl)CCC(C)C1)N(CCN(C(CC(C)P(C)(C)=O)=O)C)C 28473,C(=O)(CS(=O)(=O)CC(C)C)N1CCN(C(CC2(CC=C)CCCC2)=O)C(CO)C1 28474,Cc1ccccc1-n1cc(C(N2CC(NC(C3CC3C(=O)O)=O)C2)=O)nn1 28475,CCN=C(NCc1ccc2c(c1)OCO2)N1CCC(O)CC(C)(C)C1 28476,N1(C(C23C(CN(Cc4cccc(N(C)C)c4)C2)C3)=O)CC2CCCC2C1 28477,c1(CC(=O)N(CCC(C)NC(=O)CCCCN(C)CCO)C)ccc2c(c1)CCO2 28478,c1(C(=O)NCC2CCC(NC(CCCOC(C)C)=O)C2)ccc(C(F)(F)F)cc1 28479,N1(C(c2c(C)n(C)nc2)=O)CCCC2(CCN(C(c3cc(N)cc(O)c3)=O)C2)C1 28480,C1(NC(c2n(CC)nnc2)=O)CC2CN(C(c3cccc4c[nH]nc34)=O)CC2C1 28481,C1(CNC(COC2CN(C(C3C(C(C)C)C3)=O)C2)=O)CCCCC1C 28482,C1(OC)CC(CNC(C23CC(C2)C3)=O)N(C(=O)C(C)CC2CCCCC2)C1 28483,N1(C(c2c(CC)con2)=O)CC(NC(c2ccc(C)nn2)=O)CC1C 28484,N1(C(C(N2CCP(C)(=O)CC2)C)=O)CC2CCC1C(NC(=O)CS(C)(=O)=O)C2 28485,C1(NC(CCCOC)=O)CS(=O)(=O)C2CN(C(C3CC4CC3CO4)=O)CC12 28486,C(=O)(C(CO)C(C)(C)C)N1CC(C)C1C(=O)NCCCc1nnnn1C 28487,c1(COC)nc(N2CCC(C(C)NC(C3CC3C)=O)C2)cc(O)n1 28488,C1(N(C(C(C)c2cccs2)=O)C)CN(C(C2CC(=O)C23CCC3)=O)CCC1O 28489,CCCC(O)C(CO)NC(=O)C(CCC1CCC1)NC(=O)Cc1cccn1C 28490,CC1=CCCN(C(C2CC(=O)CN2C(C2CC(O)C(F)C2)=O)=O)C1 28491,N1(C(C(COC(C)C)NC(C)=O)=O)CCC(C(=O)NC2(C(C)O)CCC2)C(O)C1 28492,c1(C2(C(=O)NC(CNC(C3C4COCC34)=O)CO)CCCC2)cc(F)cc(F)c1 28493,N1(CC=CC(=O)NCCOCCCN(C(C2(COC)CC2)=O)C)CCCC1 28494,c1(C(=O)NCC(C2CCCC2)NC(c2cnn(C)c2Cl)=O)c(F)cc(Cl)cc1F 28495,N1(C(C(CC=CC)C)=O)CCN(C(c2cc(C)n(CC(F)(F)F)n2)=O)CC1CF 28496,O=C1NCC2(CO1)CN(C(N1CCCOC(c3ccccc3)C1)=O)C2 28497,C1(NC(C2(CNC(=O)CC3CCSC3)CC2)=O)CCN2CCCCC12 28498,CCCC(CC)C(=O)NCC1(F)CCCN(C(c2cc(O)ccc2Br)=O)C1 28499,N1(C(c2c(CC)nc[nH]2)=O)CCC(CO)(CNC(c2ccccc2C(F)F)=O)C1 28500,N1(CC(=O)NC2C(C)CN(C(C3CCCC34CCC4)=O)C2)C(=O)NC(C)(C)C1=O 28501,N1(CCNC(C(C)CC2CC2)=O)CCC(NC(C2CCOC2(C)C)=O)CC1 28502,Cc1nn(C)cc1C1CCCN1C(C1CCCCN1C(=O)Nc1ccccc1)=O 28503,c1(C(C(=O)NCc2cc[nH]n2)N(C2CCOC2)C2CC2)ccc(Br)cc1 28504,C(C(C)(C)CN=C(NCC1(c2ccccc2C)CC1)NC1CCS(=O)(=O)C1)OC 28505,C(C)(C(C)C(=O)N(C)CCc1noc(C)n1)NC(CSCCOC)=O 28506,C1(C(=O)OC)CC(C)(NC(c2ccc(CNC(c3cn(C)cn3)=O)o2)=O)C1 28507,Cc1ccc(CN2CCC(CNC(c3ccn(C4CCCC4)n3)=O)C2)o1 28508,c1(C(=O)NCC(C)CNC(=O)CNC(C2CCCC2)=O)coc(Br)c1 28509,CC(C)CC(C(=O)NC(Cc1cnc[nH]1)C(=O)NCCC(C)(C)N(C)C)C(N)=O 28510,C12(C(N(C)CC)=O)CC(CN(C(c3cnn4c3CCC4)=O)C1)C2 28511,CCCC(C)(CC)C(=O)NC(C)CCNC(=O)C1=CSCS1 28512,c1(C(N2C(CN(C(=O)C(C)O)CC)CCC2)=O)cc(C2CC2)oc1C 28513,C12(CC(=O)N(C3CC(NC(COC(C)C)=O)C3)C)CCC(CC1)CC2 28514,C(CC(=O)N1CCN(C(c2ccc(O)nn2)=O)C(C(F)F)C1)(C(F)(F)F)OC 28515,C1(CC)(CC)CC(C(N2CC(N(C(=O)C(C3CCCOC3)OC)C)C2)=O)C1 28516,C1(NC(C2C(C)C2)=O)CN(C(C2(C)CCN(CC(F)F)CC2)=O)CCC12CCC2 28517,CCCC(C)CCCC(=O)NC1CN(C(c2nnc(S)n2C)=O)CC1C1CC1 28518,C(C)(C)(CN=c1[nH]c2ccccc2o1)NC(C(C(CC)C)O)=O 28519,c1(CSCC(=O)NCCN(C(C2CCC(CO)CC2)=O)CC)ccc(C#N)cc1 28520,c1(C(N(CC(C)NC(C2CC(CN(C)C)C2)=O)C)=O)cccc(C2CC2)c1 28521,Cc1cncc2cc(C(=O)NC3CCCC3NC(C3CC(=O)NC3(C)C)=O)sc12 28522,N1(C(CN(C)CC)=O)CCC2(C=C(C(=O)NC3CC(CSC4CC4)C3)C2)C1 28523,CCCC(CNC(C1CCCC1O)=O)C(=O)NCCC1CC1C 28524,N1(C(Cc2c(C)n(C)nc2)=O)CCC(C2CC(NC(C3(C)CCCS3)=O)C2)CC1 28525,CC1CC(CCNC(=O)CCOC2CC2)CCN1C(=O)CC(Cl)Cl 28526,Cc1cc(C(=O)NCC2(C(=O)NCCCN3CCCC3C)CC=CC2)ncc1F 28527,CC(C)CC(F)(F)C(=O)NC1CCCCC1NC(=O)COC1CCOC1 28528,C1(NC(C(CCCCC)O)=O)CCN(C(c2ncc(C)cn2)=O)CC12CCC2 28529,C1(CNC(c2coc(CO)c2)=O)OCCC1C(=O)NCCCC1CCOC1=O 28530,CC1CCC(CNC(=O)CCSCC(N)=O)CN1C(c1ccc([N+](=O)[O-])[nH]1)=O 28531,c1(OC)ccnc2c(NC(=O)Cc3csc(=NCc4cocn4)[nH]3)cccc12 28532,C(=O)(C(C)(O)C(F)(F)F)NCC(CC(C)C)(C)NC(=O)CCn1cnnn1 28533,N1(C(C2C(CC)OCC2)=O)CCN(C(=O)CSCc2ccccn2)CC1CCO 28534,CC(C)C(CNC(c1cc(Cl)on1)=O)NC(C1(CO)CCCO1)=O 28535,Cc1ccc(N)c(C(=O)NCC(C)(C)NC(=O)C(C2CCCCC2)F)c1 28536,C(CNC(=O)Cn1cc(C)cn1)(CC(=O)NCCn1nncc1C)OC 28537,c1(C(=O)NCC(CCNC(C2(C)CC3CC3C2)=O)O)ccc2oncc2c1 28538,c1(OCC(=O)NC)cc(CN2CCC(CO)CC2)ccn1 28539,N1(C(C=CCN(C(C2(OC(C)C)CCC2)=O)C2CC2)=O)CCC12CCCC2 28540,N1(C(C(C)(C)OC(C)=O)=O)CCCC(C(N2CCC(N3CC=CC3)C2)=O)CC1 28541,c1(C(=O)NCC(CCOC)NC(=O)Cn2cccc2)ccn(C(C)C)c1C 28542,Cc1cccc(C(O)C(=O)NC2CC2NC(=O)CCC2(C)CC2)c1 28543,C1(C(=O)NCC2(CO)C(C)(C)C2)CN(C(C2C3CCCCC23)=O)CC1(F)F 28544,C(=O)(C(C)(C)C(C)O)N(CCNC(C1CC1c1ccnn1CC(C)C)=O)CC 28545,CCC(N=c1[nH]c(N2CCC(CO)CC2)nc2ccc(OC)cc12)c1nccs1 28546,Cc1csc(=O)n1CC(=O)NCC1CC(C)N(C(=O)C=CC(C)(C)C)C1 28547,CCC(C)CC(=O)C(=O)N1CCC2(CC(C(N3CCOC(C)C3C)=O)C2)C1 28548,c1(N(C(CN(C2CCCN(C(C(C)C)=O)C2)C)=O)C(C)=O)ccc([N+](=O)[O-])cc1 28549,C1(C)(C(=O)NC(CCCNC(C(C2CCC2)OCC)=O)C)COC(=O)N1 28550,Cc1n[nH]cc1CNC(C1OCCC1CNC(C1(C)CCC1)=O)=O 28551,n1(CC(=O)NC2(CNC(=O)COC3CCCCCC3)CC2)nnc2c1CCCC2 28552,C1(CC)CN(C(c2ccc([N+](=O)[O-])s2)=O)CCN1C(C1CCN(C)CC1)=O 28553,C(=O)(C1=CCCOC1)NCC(C1CCCC1)NC(C1(CCC=C)CC1)=O 28554,C=CCCC(F)(F)C(=O)NCCCC1CN(C(c2cnn(C(F)F)c2)=O)CCO1 28555,c1(C(=O)NCC2C(NC(c3c(OCC)cccn3)=O)C2)cc2cc(O)ccc2[nH]1 28556,c1(C(N(C2CCN(C(=O)CSC3CC3)C2)CC#C)=O)cc(Cl)n(C)n1 28557,N1(c2nc(CC)nc(Cl)c2CC)CC(NC(=O)C(O)C(C)C)C2(CCOCC2)C1 28558,C1(C(N2CCC(c3cccc(Br)c3)CC2)=O)CC2CC2N1C(C1CC1F)=O 28559,Cc1nn(C)c2ncc(C(=O)NCCOC(=O)Nc3ncc(Cl)cc3Cl)cc12 28560,c1(SC)ccc(CC(=O)NC2CCCC(NC(=O)Cc3ccc(Cl)cn3)C2)cc1 28561,C1(O)(CCNC(C(COC)OC)=O)CCCN(C(=O)CCC(C)(C)OC)C1 28562,c1(C(N(C(CN(C(C(CC=C)CC)=O)C)C)C)=O)cccn2nccc12 28563,C1(C(C(=O)NCCC(C)N(C(=O)CC2(C)CC2)C)OCC)CC(F)(F)C1 28564,C(CC(=O)NC1CCCN(C(=O)C2CC2)C1)(C(N)=O)N(C(=O)CN1CC2CC2C1)C 28565,c1(OC)cnc(Cl)c(NC(C2CCN2Cc2ccc(C(C)(C)C)cc2)=O)n1 28566,c1(CN2C(C(=O)NC3(C(=O)OC)CCC3)C=CC2)cc(O)c(Br)cc1O 28567,c1(C(=O)NC2(c3c(C)cccc3)CCC2)cccc2nscc12.n12cc(nn1)C2 28568,C(=O)(CC(F)(F)F)NC(C)C(=O)NC1(CNC(=O)CC2(C)CCCC2)CCOC1 28569,c1(C(=O)NC2CC(CCNC(C(CCC)C)=O)C2)cncc(N)c1C 28570,c1(OC)cc(C(=O)NC(CNC(C2CC(=C3CC3)C2)=O)C2CC2)c2occc2c1 28571,C(=O)(CC(O)c1ccccc1)NCCC(C)N(C)C(C1(C)CCCC1)=O 28572,CCC(C(=O)N1CC(CN(C)CC)C1)N(C)C(C1CC(CC(=O)OC)C1)=O 28573,c1(C(N2C3C(NC(CSCC#C)=O)CC(C3)C2)=O)cccc2nccnc12 28574,c1(C(=O)NCc2ccsc2C(N2CCC2)=O)n[nH]cc1[N+](=O)[O-] 28575,C(=O)(C(F)(F)F)NC(C(C)N(C(C)=O)NCCCN(C1COC1)C1CC1)=O 28576,CCC(C(=O)NCC1CN(C(c2ccc(C(C)C)cc2)=O)CC1(F)F)C(C)C 28577,c1(NC(C)=O)c(C(N2CCC(NC(=O)Cn3cccc3)C2C)=O)cccc1C 28578,C#CC1CN(C(=O)CCc2cn[nH]c2)CCN1C(c1cnc(O)o1)=O 28579,CN1CCC(C(=O)N2CC(CO)(NC(=O)C3=CCCC3(C)C)C2)c2ccccc21 28580,c1(C(N(C)CC2C3CN(C(CN(C(C)=O)C)=O)CC32)=O)ccc(F)c(C(F)F)c1 28581,C1(N2CCOCC2)(CNC(=O)Nc2nc(N(C(C)=O)CC)sc2)CCN(C)CC1 28582,N1(C(C2(C(C)C)COC2)=O)CCOCC(NC(=O)C(C)Oc2ccccc2)C1 28583,C1(CNC(CC2CC(C(=O)OC)C2)=O)CCCCN1C(=O)COCP(C)(C)=O 28584,N1(C(CCC=C(C)C)=O)CCOC2(C1)CN(C(=O)C(C)Oc1ccccc1)C2 28585,CC1CCC(C)(C(N2CC3(CC(NC(c4[nH]cc5c4CCC5)=O)C3)C2)=O)CC1 28586,Cc1ccnc(O)c1C(=O)NCCC1CC(N)C1 28587,S(=O)(=O)(c1ccc(C)c(C)c1)N1C2(CNC(C(CCCC)O)=O)CCC1CC2 28588,C1(NC(c2c(CC)oc(C)c2)=O)C2CC3C1C3C2C(N1CCC1C(C)(C)O)=O 28589,CC1CN(C(c2sccc2CNC(=O)CCc2cccn2C)=O)CC1O 28590,Cc1ccc(O)c(CC(N2CCN(C(c3nc(O)sc3C)=O)C(C)C2)=O)c1 28591,CC1CCCCCN1C(=O)CCOCCNC(c1cncc(F)c1)=O 28592,N1(C(c2cccc(N3C(=O)CCC3)c2)=O)CC2(C(=O)O)CCC2(C(=O)O)C1 28593,c1(C(=O)NCC2(CNC(C(c3cncnc3)C)=O)CCC2)ncc(Cl)cc1F 28594,C1(C(N(C)CCNC(C2CCC(C(F)(F)F)CC2)=O)=O)CCc2nnc(O)n2C1 28595,C1(C(N(CC)CC2CCOC2)=O)CC2CN(C(=O)CN3CCCC3=O)CC2C1 28596,C1(C)(NC(CC2OCCN(C(C3CCN(C)CC3)=O)C2)=O)CCC(C)(C)C1 28597,CCC(CCCO)NC(=O)C(CO)NC(=O)CC(C)=C(C)C 28598,c1(CC(=O)NC(CC2CN(C(c3cc(C)oc3)=O)C2)C)cnc(Cl)cc1C 28599,C1(O)(CC(=O)N(C(C)CNC(=O)C(c2ccc(Cl)s2)C)C)CCCCCC1 28600,CC1=C(C(=O)N2C3CCC(C3)C2CC(N2CC(F)(F)CC2CO)=O)CCC1 28601,c1(C(=O)NC2CN(C(CC3CC(C)(C)OCC3)=O)C2)cc(F)cc2nn[nH]c12 28602,C1(NC(c2nnc(C)s2)=O)C2CC1CN(C(C1CC1C1CCCC1)=O)C2 28603,C(=O)(C(C)(C)CS(N)(=O)=O)N1CC2C(CNC(c3ccc(COC)cc3)=O)(C2)C1 28604,C(c1cccc(Br)c1)=CC(=O)NCCCCN(C)C(C1(C(N)=O)CC1)=O 28605,c1(C(C2CCOC2(C)C)NC(=O)NC(CCOC)c2cccs2)cc(C)ncc1C 28606,CC1(C(=O)N2CCC(NC(=O)COc3cn[nH]c3)C2)COc2ccccc21 28607,C(=O)(CCS(=O)(=O)CC(C)C)N1CC(NC(Cc2cc(C)on2)=O)C(CO)CC1 28608,c1(C(=O)NC(CC=C)CNC(c2cnc(C(F)F)nc2)=O)cc2n(n1)CCC2 28609,CC(Cc1cccn1C)N=c1ccnc(NC2CCC(=O)NC2)[nH]1 28610,N1(C(C2(C#N)CC2)=O)CCC(O)C2(CCN(C(=O)CCC3CCCC3)CC2)C1 28611,c1(C(=O)NC2CC(NC(c3ccn(C(C)C)n3)=O)C2)ccc(=O)n(C2CC2)c1 28612,CC(=NO)C1CC(C(N2CC(NC(=O)CSCc3ncc[nH]3)C2)=O)C1(C)C 28613,Cc1cccnc1C(=O)NC(C1CCOC1)CNC(c1cncc(C(F)F)c1)=O 28614,N1(C(c2c(CNC(CC=CC=C)=O)n[nH]c2)=O)CCc2ccncc21 28615,Cn1nc(C(=O)NC2CC2NC(C2CC3(CC3)CO2)=O)cc1C1CC1 28616,c1(SC)ccc(Cl)c(C(N2CCN(C(=O)CC3CC4(CC4)CO3)CC2C)=O)c1 28617,c1(C(N(C(CN(C)C)(C)C)C2CC2)=O)ccccn1.C1CC(=O)N1 28618,C1(C(N(CCCNC(=O)C(O)P(C)(C)=O)C(C)C)=O)CCn2nccc2C1 28619,c1(C(C)(C)C)ccncc1C(=O)NC1CCCC(NC(C2CC2F)=O)C1 28620,c1(C(=O)NCC23C(CN(C(CC=CCC)=O)C2)C3)ccc(F)c(C(F)(F)F)c1 28621,C1(C(=O)OC)CC(SC)CN1C(=O)CC(C)(C)c1cn(CCSCC(C)C)nn1 28622,c1(C(=O)NCC2N(C(CC(C)C)=O)CC(C)CC2)cccc2cc[nH]c12 28623,C(CC(=O)N1CC(N(C)C(C23CCC(C)(CO2)C3)=O)C1)(C(C)C)OCC 28624,c1(-n2ccc(C)n2)ccccc1C(=O)NCC(F)CNC(C1CCOCC1)=O 28625,C1(C(=O)NCC2C(NC(c3cc(C(F)(F)F)ccn3)=O)CC2)CC2(CCCC2)C1 28626,N1(C(Cc2cncc(C)c2)=O)CC(F)(F)CC1CNC(c1nc(C)ccc1C)=O 28627,c1(C(N(CCN(C)CC2CCC(C)(C)CC2)C)=O)occ2c1CCC2 28628,N1(C(C=CC(C)(C)C)=O)CC(NC(=O)C=C2CCCCC2)C2CCCC12 28629,c1(C(=O)NC2CC(NC(C3C(C)(C)COCC3)=O)C2)ccc2cc[nH]c2n1 28630,O=C1CC(C(=O)NCCNC(=O)C2=CC3(CCOCC3)C2)c2cccnc2N1 28631,C(C(=O)N(CC(C)(O)C1CC1)C)(C(C)OC)NC(CC1(CSC)CC1)=O 28632,CC1(CC(=O)Nc2ccn(C3CC3)n2)CCN(C(=O)CCCn2cccn2)C1 28633,c1(NC(=O)OC)snc(C)c1CSC1CCN(C(C2CCCN2C)=O)C1 28634,C1(CC)CCC(C(=O)N(C2(C(N3CC(C(F)(F)F)C3)=O)CC2)C)CC1 28635,C1(CNC(COCC(=O)NC)=O)CN(C(=O)CCc2ccc(NC)cc2)CCO1 28636,c1(C(N(CCN(C(C(C(=O)OC)OC)=O)C)C)=O)ccc(C(F)F)c(C)c1 28637,C1(C(=O)OC(C)(C)C)CCC(C(=O)O)CC1.n12cc(nn1)CNC1CC2C1 28638,n1(COC)ncc2cc(-c3ccc(NC(N4CCOCC4)=O)cn3)cnc12 28639,CCC(C(C)(F)F)C1CCN(C(=O)CCCOCCN)CC1 28640,C#CCCCCC(=O)NC1CCC(CNC(=O)CC2CCCS(=O)(=O)C2)CC1 28641,N1(C(C2(OCC)CCC2)=O)CCCCC1CNC(=O)C(c1cccc(F)c1)O 28642,Cc1cn2cc(C(N3CCN(C4CN(C(=O)C=CS(C)(=O)=O)C4)CC3)=O)sc2n1 28643,C1(C(=O)NC(C=C)CO)CCCCN1C(c1cncn1C1CC1)=O 28644,c1(C(=O)NCC(CN(C(C(C)N(C(C)=O)C)=O)C)(C)C)cccc(CS(C)=O)c1 28645,C1(CC(=O)OC)CN(C(CC2CCC3CC23)C(=O)NC2CC2)CC(C)O1 28646,CC1(C)CC1(S(C)(=O)=O)C(=O)OCc1cc(Br)cc(I)c1 28647,Cc1cnc2cc(C(N3C4CCC3C(CNC(=O)COCC(C)C)C4)=O)ccn12 28648,c1(C(=O)NCC(c2ccc(OC)cc2)O)c[nH]c2cc(-c3nn[nH]n3)cnc12 28649,C(=O)(CC(C(F)F)C(C)(C)C)NCCN(CCCc1cccc(OC)c1)CC 28650,c1(C(=O)NC(C2CCCN(C(COCC(=O)NC)=O)C2)C)c[nH]c(=N)nc1C 28651,C1(C(=O)NC2(CO)CC(CO)C2)(CNC(C2C(OC)CCC2)=O)CC12CCC2 28652,C1(C(=O)NC(C)(C)CNC(c2[nH]ccc2-c2ccccc2)=O)CCC2(CCC2)O1 28653,C(C)(C(=O)N(C1CCC1)C(C)CO)N(C(=O)C=CCF)CC 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28776,CCCC(F)C(=O)NC(COC)CC(=O)NCC1(CN(C)C)CCC1 28777,Cc1nnc(O)c(C(N2CC(NC(=O)CCCN=[N+]=[N-])C(C)C2)=O)c1C 28778,N1(C(C(C=CC)O)=O)CCC(CO)(CNC(C2(OC)CCC(C)(C)C2)=O)CC1 28779,C=CCCCC(=O)NCCOCCNC(c1cnc(SC)n1C)=O 28780,c1(C(C)NC(N2CC(CO)OC(C3CCCCC3)C2)=O)cnc2n1CCCC2 28781,C1(CNC(CC2C(C)C2)=O)COCCN(C(c2ccc(CC3CC3)s2)=O)C1 28782,c1(C(=O)NCC(CNC(c2cc(C)no2)=O)S(C)(=O)=O)ccn2ncnc2c1 28783,C(=O)(C(O)C(C)(C)C)NC(C)CC1CCN(C(c2cc(C(C)(C)C)no2)=O)CC1 28784,C#CCS(=O)(=O)CCNC(=O)NC1(C)CC=CCO1 28785,C(=O)(C(=O)C(C)(C)C)NCC1(OC)CCN(C(=O)CCn2ccccc2=O)C1 28786,C1(CNC(CCC2CCC(C)O2)=O)CN(C(c2coc(C(F)F)n2)=O)CC1(C)C 28787,c1(NC(C2CC(NC(CNC(CCC)=O)=O)C2(C)C)=O)n[nH]c2ccccc12 28788,c1(OC)nn(C)cc1C(=O)NCC12CC(CN1C(c1csnn1)=O)C2 28789,C(=O)(C(O)(C(C)C)C(F)(F)F)NC1CN(C(CCn2c(C)ncc2)=O)C(C)(C)C1 28790,CCC(C(=O)N1CCN(C(=O)C=CC2CCOCC2)CC(C)C1)C(F)(F)F 28791,N1(C(c2cc(CCC)[nH]n2)=O)CC(C)(CNC(=O)CS(=O)CC)CC1(C)C 28792,c1(C(=O)NCC(=O)NC(C2CCCCO2)CC)ccc2[nH]nc(Cl)c2c1 28793,N1(C(COCC(=O)N(C)C2CC2)=O)CC2CC(O)C1C2NC(=O)CN1CCCCC1 28794,N1(C(C2N(C)CCC2)=O)CCCC2(CCN(C(c3cnn(C)n3)=O)C2)C1 28795,C(=O)(C1=CCCCO1)NC1C(C)(C)C(CC(=O)Nc2ccc(C3CC3)nc2)C1 28796,c1(C(=O)NC2C(NC(C3(C(=O)OCC)CC3)=O)C2)occc1C 28797,N1(C(C2C3COCC23)=O)CCCC(C(=O)NC(c2ccccc2F)CO)(CO)C1 28798,C(=O)(CCC(C)(C)[N+](=O)[O-])N1C(C(N2CC(N(C)C3CC3)C2)=O)CCC1C1CC1 28799,C12(CNC(COCCCC)=O)CCN(CC1)C2.c1(CC)nc(CC)ns1 28800,c1(NC(CN(C(=O)C(CC)=CC)CC#C)=O)ccc(N(C)C)cc1 28801,C(=O)(C(CC(C)C)N(C)C(c1cc(C(N)=O)[nH]n1)=O)NCc1[nH]nc(CC)n1 28802,N1(C(C2(C)CCN(S(=O)(=O)C3CCCCC3)C2)=O)CCc2ccc(F)cc2C1 28803,C(=O)(C(C(C)(C)C)c1ccccc1)N1CC(OCCNC(c2cn(CC)nc2)=O)C1 28804,C(=O)(CC(C)C(C)(C)C)N1CC=C(C(=O)NC(C(C)(C2CC2)NC(C)=O)=O)C1 28805,Cc1nc2ncc(C(N3CC4C(NC(C5CC(C)(C)CO5)=O)C4C3)=O)cc2o1 28806,C1(NC(CC2CC(=O)C2)=O)CC(O)C1NC(=O)COCC1CCOC1 28807,c1(CCC(=O)NC2C3CCC2N(C(=O)Cn2ncnn2)C3)csc2ccccc12 28808,N1(C(c2c(C(=O)OC)coc2)=O)CCN(C(c2n[nH]c3c2CCC3)=O)C2CC12 28809,CC(C)CS(=O)(=O)CC(=O)N1CC(O)CC1CNC(c1ccccc1)=O 28810,C(=O)(CCC(c1ccccc1)N(C)C)N(C1CCN(C(=O)C(C)(C)F)CC1)CC 28811,CC1(C)CC(C(=O)NC2CC(NC(c3ccc(O)nc3Cl)=O)C(O)C2)CCO1 28812,N1(C(=O)NCCCC#C)Cc2nnc(C)n2CC1C(=O)OC 28813,c1(C(=O)NCCN(CCC)C(c2cccc(CF)c2)=O)nn(C)c2c1CCC2 28814,N1(C(CSSC)=O)CCN(c2cc(CNC(=O)CCC(F)F)ccn2)CC1 28815,n1(CCNC(=O)C(O)Cc2cnc[nH]2)cc2ccccc2n1 28816,CCC(C(=O)NC(c1cccnc1)C(=O)NCCn1nncc1C)n1ccnc1 28817,C12(CNC(=O)CC3CCCO3)CN(C(=O)C=CSc3ccccc3)CC(F)(C1)C2 28818,CC(C)CC(C(=O)NC(CO)CC(C)C)NC(C1C2CCC(F)C12)=O 28819,C1(C(N(CCCNC(C2CCN(C)C2)=O)CC)=O)CC12CC(C)(C)C2 28820,CN1CCCC1CCC(=O)NC(CC1CCC1)C(=O)NCC1CCN(C(N)=O)C1 28821,N1(C(C2C(CNC(c3c(C)nc(O)cc3)=O)CCC2)=O)CC(C)C12CCOCC2 28822,c1(NCC(c2c(C)n[nH]c2)C)ccc(SCC2CCCO2)cc1 28823,N1(C(c2c(OC)nccc2)C(=O)Nc2ccc(F)cc2)CCCC(C)(O)CC1 28824,CC(Cl)(Cl)C(=O)NCC(C1CCOC1)NC(=O)C=Cc1cc[nH]n1 28825,C1(CNC(C(COCC)C)=O)CN(C(=O)Cc2cccnc2Cl)CC1O 28826,c1(CC)nc(C)c(C(=O)NC2CCC2NC(c2cn(CC(N)=O)nn2)=O)s1 28827,CCCC(C(=O)NCc1cc(C(N2CCC23CC(C)(CO)C3)=O)ccn1)C(C)C 28828,c1(C(=O)NC(CN(C(c2cc(C)[nH]c2)=O)C)C)cc(C#N)ccc1C 28829,c1(CN(CC=C)C)cc(C)c(-c2ccccc2OC)s1 28830,c1(C(N2CC(CC(C)NC(CCCNC(C)=O)=O)C2)=O)ccc(C(N)=O)cn1 28831,C1(NC(CSCC#C)=O)C(CNC(c2cc3ccncc3s2)=O)CCC12CCC2 28832,c1(OCC)ccc(Cl)c(C(=O)NC23CC(C2)N(C(C2CCCCC2OC)=O)C3)n1 28833,N1(C(C2(CCC)CC2)=O)CC(NC(=O)Cc2ccccc2O)CC(C)(C)C1 28834,C1(C2CCC2)(C(=O)NCC2N(C(=O)Cc3ccccc3F)CC2)CC1(F)F 28835,c1(C(c2nnnn2C)NCCS(N(C)C)(=O)=O)ccc2c(c1Cl)OCCO2 28836,N1(C(c2[nH]cc(CC)c2)=O)CC(CNC(=O)CC2C(C)(C)C2(C)C)C2(CC2)C1 28837,C1(c2nnnn2C(C)C)(NCCC2(SC)CCCC2)CCCC2CC12 28838,C(=O)(C(F)C(C)CNC(c1cc(C)cc(O)c1)=O)NC(COC)(C)C 28839,CCC(C(=O)NCCC1(OC)CCC1)NC(=O)Cc1n[nH]c(C)n1 28840,Cc1cc(F)cc(C)c1C(=O)NCC(C)CNC(C1CN2CCN1C(C)C2)=O 28841,C=CCCCCCN(C(=O)CC1CCCN1C(=O)C(O)C1CCC1)C 28842,C(CCCCC(=O)N(CCCCN(C)C(C1CCCN(C(C)C)C1)=O)C)OC 28843,C1(NC(C(CCSC)O)=O)CCC2(CCN(C(C3(CCN(C)C)CC3)=O)C2)C1 28844,Cc1cccc(C(=O)NC2CCCCC2NC(=O)COc2ccsc2)c1F 28845,C1(O)(CC(=O)NC2(CF)CCN(C(c3c(C(C)C)ocn3)=O)C2)COC(C)(C)C1 28846,O=C(C1=CCCO1)NCC(C1CCCC1)NC(=O)C(F)(F)c1ccccc1 28847,c1(-c2nnc(N3CC(C)(C)SCC3)n2Cc2ccccc2)ccc2ccoc2c1 28848,N1(C(CCc2n(C)ccn2)=O)C(C(=O)NC2CCOC2)CC2CCCC12 28849,c1(C(C(=O)N(C2CN(C(C3C(OCC)C3)=O)C2)C)C)cccc(Cl)c1 28850,C1(NC(CCC)=O)CCC(C(=O)NCc2cccc(C(C)(C)C)c2)CC1 28851,c1(NC(C2C(NC(C3CN(C)C3)=O)CCC2)=O)cc(C(F)F)cnc1Br 28852,C(=O)(CCCCCNC(C1(C(=O)NC2CC2)CC1)=O)N(CC(CN(C)C)O)C 28853,c1(-c2c(C)ccc(CO)c2)cncc2sc(C(=O)Nc3cnn4c3CCC4)cc12 28854,c1(OC)c(CCC(N2CC(CC(C)NC(C3CCC3OC)=O)C2)=O)cccc1Br 28855,C1(NC(c2sccc2C#N)=O)CCC(O)CN1C1(CCCC)CC1 28856,C(=O)(N=c1[nH]oc2c1CC(C(C)(C)C)CC2)c1nn(C)nc1Br.c12nc(cs1)C2 28857,C(CCC(C)(C)NC(C1CSCN1C(=O)C(C)OCCN(C)C)=O)OC 28858,C12(NC(C(C)Sc3ncccn3)=O)CCCCCC1N(C(=O)CC(C)(F)F)CC2 28859,N1(c2nnc(C#N)s2)CCC2(NC(=O)CCc3ncc(F)cn3)CCCC12 28860,Cc1cc(C(N2CC3CC(CNC(c4cnc(O)o4)=O)C3C2)=O)n2nccc2n1 28861,c1(CNCc2c(OCCCC)nccc2)nc(Cl)c(C)cc1F 28862,N1(C(C(C)N(C(C2CCCCCN2C)=O)CC)=O)CC2CCCCC12C 28863,C1(c2n(CC)nnn2)(NC(c2ccc(SC)cc2)C)CCCC2(CCCCC2)C1 28864,C(C(=O)NCC1CCC(F)(F)C1)(C(C)(C)C)NC(c1c(CC)cno1)=O 28865,C1(c2nc(C3(CN)CCCCO3)on2)CC12CCOc1ccccc12 28866,N1(C(=O)CCc2ccc(O)cc2)CCC2CCCC12CNC(C1(F)CCCC1)=O 28867,C1(CC)CC(C(N2CCSC3CCC23)=O)CCN1C(=O)C(F)C1CCCC1 28868,C1(NC(C(C)N(CCC)C(c2cc(O)cs2)=O)=O)CCC2CCC12 28869,C1(NC(c2cc(C3CCC3)no2)=O)CCN(C(c2nc(Cl)c(Cl)s2)=O)CC1O 28870,c1(C(=O)NCCC2CC(NC(C3CCC3)=O)C2)cnoc1-c1ccccc1 28871,c1(C(=O)NCC2CC(NC(C(C)=C3CCC3)=O)CC2O)ccnc2c1ccn2C 28872,c1(CNC(CC(=O)NCCCC)Cc2cccs2)cccc(F)c1I 28873,C1(CC=C)(NC(=O)CS(=O)(=O)CCO)CC2CCC(C1)N2C(=O)C(C)CF 28874,C1(OCC)CC(NC(C2CC23CCC(F)(F)CC3)=O)C12CCCCC2 28875,C(=O)(C1=CC2(CCOCC2)C1)NCC(C(C(C)C)C)NC(c1c[nH]ccc1=O)=O 28876,N1(C(c2ccc(N)c(Cl)c2)=O)CCN(C(=O)Cn2ncnn2)C2CCCCC2C1 28877,N1(C(CC(=O)OC(C)(C)C)=O)CC(C(=O)NCC(F)CO)CC12CCC2 28878,C1(O)(CCNC(c2c(CC)c[nH]n2)=O)CCCN(C(C2CCCC2CC)=O)C1 28879,CCCCC(C(=O)N1CC2CCC2(CNC(=O)Cc2cccc(Cl)c2)C1)N(C)C 28880,c1(C(N(C2CCC(NC(CCC(=O)N(C)C)=O)C2)C)=O)oc2ccccc2c1Cl 28881,c1(C(c2cnsc2)NCC(n2ccnn2)C)nnnn1C1CCCCC1 28882,C#CCC(C(=O)N1CCCC(CCNC(c2cnn(C3COC3)c2)=O)C1)C1CC1 28883,C12(C(=O)NC3C(C)(NC(C4C(CC)CCO4)=O)CCC3)CC=CCN1CCC2 28884,N#Cc1cccc(-c2cn(CCCCNC(=O)Cc3nc[nH]n3)nn2)c1 28885,C1(CC(=O)NC(CCCNC(c2c(CC)nco2)=O)C)CCC(F)(F)CC1 28886,C(=O)(CCCC(F)(F)F)NCC(C)NC(C(c1ccc(OC)cc1)C)=O 28887,C(=O)(C1CCCc2nn(C)cc21)NCC(C)NC(=O)CCc1c(F)cccc1Cl 28888,C1(F)(C(N2CCN(CCCCCNC(C=CCC)=O)CC2)=O)C2CCCCC12 28889,Cc1cc(C(=O)NC2CN(C(=O)Nc3cccc(CO)c3)C2)cc(NC2CC2)n1 28890,c1(C(C(=O)NCCN(C(=O)C(=O)N(C)C)CCOC)C)cn(C)c2ccccc12 28891,N1(C(C(C)OCCC(C)C)=O)CCC(C(N2CC3CCC(C2)N3C)=O)C12CCC2 28892,Cc1ccnnc1C(=O)NCC(C)N(C(=O)C#CC(=O)N(C)C)C 28893,N1(C(c2c(NS(C)(=O)=O)nccc2)=O)CC2(CC(NC(=O)C3=COCCC3)C2)C1 28894,C(CNC(c1ncsc1C(F)(F)F)=O)(C(C)C)NC(C1CC(N(C)CC)C1)=O 28895,C1(C(=O)Nc2cc(CCC)n[nH]2)COCC1(C)C 28896,CC1CCN(C(c2ccc(Cl)cc2N)=O)CC1NC(=O)CSc1ccccc1 28897,C=CC1(CNC(=O)NCCN(C)CC)CCC1 28898,C12(CNC(C(C)CC(N)=O)=O)CCC(CN(C(c3cc4cccnc4[nH]3)=O)C1)C2 28899,N1(C2CCN(CC(C)F)CC2)CCN(C(=O)CCc2cccnc2)C(=O)C1 28900,C=CCC(CC)C(=O)NCC1CC1CC(=O)NC1CNC(=O)C1 28901,N1(C(CNC=O)=O)CCC2(CCN(C(=O)CC3COC(C(F)(F)F)CO3)CC2)C1 28902,C(CCS(C)=O)(C(=O)NCC1CN(C(=O)C2=CCSC2)C1)N(C)C 28903,N1(C(C(c2cn(C)nc2)=O)=O)CC2CC(NC(C3CC4(CCCO4)C3)=O)C1C2 28904,Cc1nccc(C(=O)NC2C3CN(C(c4c(Cl)noc4C)=O)CC23)c1O 28905,C#Cc1ccc(C(N2CCN(C(=O)Cc3ccoc3C)C3CC23)=O)cc1F 28906,CC1=NOC(=O)C1CC(=O)NCC1(CNC(C2(O)CC(F)(F)C2)=O)CC1 28907,N1(C(c2c(CNC(c3cc(CC)n(C)n3)=O)c[nH]n2)=O)CC2CC1CN2C(C)C 28908,C(=O)(C#CC1CCOCC1)NC(C1CCCCC1)C(=O)NC1C(C)C1C 28909,c1(C(N2CC(C(C)NC(c3ccc[nH]3)=O)C2)C(N)=O)ccc(Br)cc1 28910,N1(C(C(N2CCCC(O)C2)C)=O)C2CCCC1CN(C(c1ccno1)=O)C2 28911,C1(C(=O)NCCN(C(CCOCCOCC)=O)CCCC)C(C=C(C)C)C1(C)C 28912,C#Cc1cccc(C(=O)NC(CCC)CCCNC(C2CC(C)(C)CN2C)=O)c1Cl 28913,N1(C(C2(CC)CC2)=O)CCC2(C(=O)Nc3ncc(Br)nc3OC)CCCC12 28914,c1(NC(c2n(CCC)nnn2)c2cccnn2)ccc(-n2nccn2)cc1OC 28915,Cc1cccc(C(N2CC(NC(=O)C(C(C)(C)C)NC(N)=O)C(C)C2)=O)c1N 28916,c1(C(=O)NC(C#C)C2CC2)cccc(CNC(C2CC3(CC3)CO2)=O)n1 28917,N1(CC(CCC)O)CCOc2cccc(OC)c21 28918,C1(CC(=O)NCC2C(NC(C(c3ccccc3)C)=O)COC2)CCC=CCC1 28919,C=C(C)CC(C(=O)N1CC(OCCF)C1)NC(=O)Cc1nocc1C 28920,C(=O)(CC(CC)c1cn[nH]c1)N(CCN(C(C(=O)NCC)=O)C)C(C)C 28921,C1(C(N2CCCC(F)(C(=O)O)C2)=O)CC2CCCCC2O1 28922,CN1CCC(O)(CNC(c2cc(CNC(C3(C)CC3(C)C)=O)cs2)=O)C1 28923,N1(C(C2(C)CCCCCC2)=O)CCC(C)(C)C(NC(C2CCCO2)=O)C1 28924,C1(Cn2c(C)ccc2C)CN(C(=O)OCCC2CC[Si](C)(C)C2)CCCO1 28925,C(N=c1[nH]c(=NCC2=CCN(C)CC2)[nH]c2c1SCC2)c1cn(CC)nn1 28926,c1(C(=O)NC2C(CNC(CC3N(CC)CCC3)=O)CC2)sc(Br)c(C)c1C 28927,Cc1cnc(NCC(C)(CC(C)C)NC(=O)CO)c([N+](=O)[O-])c1 28928,c1(OC)ccc(Cl)c(C(=O)NC2CN(C(c3cc4n(n3)CCC4)=O)C3CC23)c1 28929,C1(N(C)C(c2cc(C3CCC3)[nH]n2)=O)CCCN(C(c2cnn(C)n2)=O)C1 28930,N1(CCOC)CC(NC(=O)NCC(Cl)Cl)C(C)C1 28931,c1(NC)ccc(C(=O)NC(Cc2ccco2)C(=O)N2CCC2C(N)=O)nc1 28932,C1(CNC(c2c(C)nns2)=O)CC(C)N(C(C2CCC(NC(N)=O)CC2)=O)C1 28933,C1(C(=O)NC2C(CNC(CCCC(N)=O)=O)COC2)C2C3CC4C1C1C2CC3C41 28934,c1(SCC)ccccc1CC(=O)NCC1CCN(C(=O)CC2CC3(CC3)C2)CC1 28935,CC1(C)CCC(C(N2CCOCC2CCNC(C2COCCN2C=O)=O)=O)CC1 28936,C(=O)(CCCC(C)(C)C)NCC(C)=CC(=O)NCCC(O)C(C)C 28937,N1(C(c2nc(CC(C)C)sc2)=O)CC2CC(NC(=O)CCN3CCCC3=O)C2C1 28938,N1(Cc2cn(-c3ccc(C)c(C)c3)nn2)CCc2cc(-c3nn[nH]n3)ccc2C1 28939,C(=O)(CCC(C)S(=O)(=O)Nc1cccc(C(CC(=O)O)OC)c1)OC 28940,CCC(C(=O)NCC1(OC)CN(C(=O)CC(C)F)C1)N(C)C 28941,Cc1sc(NC(=O)C2CC2)c(C(=O)OCCSC2CCCN2C(=O)CC#N)c1C 28942,c1(-c2cn(CC(CNC(=O)C(c3cncnc3)C)OC)nn2)cc(C)ccn1 28943,C=Cc1ccc(C(=O)NC2CCC(CNC(c3ccc(CCC)s3)=O)C2)cc1 28944,CS(=O)(=O)CC(=O)NC1CCC1NC(c1cccnc1O)=O 28945,c1(-c2cc(CC)no2)nc(CCOC)nn1Cc1ccccn1 28946,Cc1cc(C(=O)NCCOC(C)(C)CNC(C2CC=CCO2)=O)sc1C 28947,C1(N(C(CS(=O)(=O)NC)=O)C)CN(C(C2CC(F)(F)C2)=O)CCC1O 28948,C1(NC(COCCC=C)=O)CC(C2CCN(C(=O)C=Cc3cccc(C)c3)C2)C1 28949,c1(CC)nccn1C(C)CC(=O)NCC1(NC(=O)CCc2ccccn2)CC1 28950,c1(C(=O)NC(C2C(C(N(C(C#C)C)C3CC3)=O)C2)C)ccc(F)s1 28951,c1(C(N(CCCN(C)C(C2CSCCS2)=O)C)=O)ccc(-n2cccn2)nc1 28952,N1(C(Cc2cncc(OC)c2)=O)CCC(NC(=O)CCc2nc[nH]n2)C(O)C1 28953,C1(n2ncc(C(N(C3CCCN(C(=O)C(C)(F)F)C3)CC)=O)c2)CCC(C)CC1 28954,c1(C(=O)NC)ccc(C=CC(=O)NCC(CO)NC(C2CCCSS2)=O)cc1 28955,C(=O)(C1=CCCN(C(C23CC(C(F)(F)F)(C2)C3)=O)C1)Nc1ccc(N(C)C)cc1 28956,CCC(CC(C)CO)NCc1cn(Cc2occc2C(=O)O)nn1 28957,C=C(Cl)C(C)(C)C(=O)N1CCC(CN(C)C(C2CC23CCCC3)=O)C1 28958,O=C(C1=CCS(=O)(=O)C1)N1CCC2(C1)CN(C(c1cc(F)cc(F)c1)=O)C2 28959,C1(NC(C(C)Oc2ccccn2)=O)CCCN(CCn2cc(Cl)cn2)CC1 28960,Cc1ccc(F)c(CC(=O)N(C)CCN(C(=O)C(c2ccccc2Cl)O)C)c1 28961,C(CCS(C)=O)(C(=O)N1CCC(OCc2ccc(Cl)c(F)c2)C1)N(C)C 28962,C(=O)(C1=CCC(C)CC1)N1CC2CC(C(=O)NC(CCCCC)C)(C1)C2 28963,C(=O)(CCCCC(=O)N(c1ccc(Br)c(C)c1)C)c1ccc(OC)cc1 28964,C1(COC)(NC(c2ccccn2)=O)CCN(C(c2ccc(C(N)=O)[nH]2)=O)CC1 28965,c1(CC(=O)NCCC2CC(NC(CCN(CCC)C)=O)C2)ccc2c(c1)CCC2 28966,C1(NC(C2CC(OCC)C2)=O)CCC2(CCN(C(C3(C)CC(C)(C)C3)=O)C2)C1 28967,C1(C(=O)NCCc2c(C)noc2C)CC(O)CCN1C(c1cnc(O)o1)=O 28968,N1(C(c2c(C)nn(C3CCC3)c2)=O)CCN(C(C2(C)CC3CC3C2)=O)CC1C 28969,CC(CCCO)(N=c1ccn(CC(F)F)[nH]1)c1nnnn1-c1ccc(F)cc1 28970,C1(CC(=O)NC(c2c(C)nccc2)C)C2CCCC2N1C(=O)C(C#N)C(C)C 28971,C1(CNC(c2ccco2)=O)(CNC(c2cc(O)cs2)=O)CC12CCC2 28972,C(c1cccc(F)c1Cl)=CC(=O)NCCC1(CNC(CCN(C)CCO)=O)CC1 28973,c1(N(C(COC(CNC(C(C2CCOC2)OC)=O)(C)C)=O)C)ccccc1 28974,c1(C(N2CC(c3c(C(N(CC)CC)=O)nco3)C2)=O)cccc(C(N)=O)n1 28975,C1(C(=O)NC2(COC)CCN(C(=O)CCCC(F)(F)F)C2)CC2C=CC1CCC2 28976,c1(Nc2c(SC)cc(C)cc2)cc2c(cc1Br)CCC2 28977,CC1CN(C(=O)CCC(=O)c2cccc(F)c2)CC1NC(C1CC1C)=O 28978,c1(NC(=O)CCNC(c2ccc(Cl)o2)CO)ccc(Cl)cc1F 28979,CC(C)CC(CCO)NC(C1OCCC1CNC(c1ccn(C2CC2)n1)=O)=O 28980,c1(C(=O)OC)cc(C)cnc1NC(C1CCCCN1C(C1CC(=O)NC(=O)N1)=O)=O 28981,Nc1cc(C(=O)NC2CCC(NC(=O)CC3CC4CC4C3)CC2)c(F)c(O)c1F 28982,c1(CC)cccc(C(=O)N(CCCNC(=O)CCSCC(C)C)CC)n1 28983,N1(CCSC)C(=O)NC(c2csc(C#N)c2)C2=C1CN(c1ccc(Cl)cc1)C2=O 28984,S(=O)(=O)(c1ccc(N2CCCC(OCC(F)F)C2)cc1Br)NCC1(C)CSC1 28985,C#Cc1ccc(Cl)c(C(=O)NC2CCCC(NC(c3cnsc3C)=O)C2)c1 28986,c1(OC)ccccc1SCC(N1CCOCC1CN(C(=O)C(C)NC(C)=O)C)=O 28987,C1(C(=O)NC2CC(CNC(C3C(C)(C)CC3)=O)C2)CCCN(CC(F)F)C1 28988,c1(NCc2c(-c3c(F)cccc3)nccc2)cccc2c(Br)cccc12 28989,C1(NC(=O)CONC(=O)CC2C=CCCC2)(CO)CCOCC1 28990,C(N=c1[nH]c(=NCC2CN(C3CCC3)C2)[nH]c2ccsc12)c1c(C)cccc1Cl 28991,c1(C(=O)NC2C(CNC(C(C)(C)c3cnc[nH]3)=O)C2)cccc(-n2ccnc2)c1 28992,N1(C(c2c(NC)nccc2)=O)CC2CC(NC(=O)Cc3cncnc3)C(C2)C1 28993,C(=O)(C1CCCc2nncn21)N1CC2CN(C(CN(C)C3CC3)=O)C2CC1 28994,N1(C(C2N(C)CCC2)=O)CCN(C(=O)C(O)C2CC2)C(CO)C1 28995,c1(C(C)C)ccc(-n2nc(COc3ccccc3)nc2C2CC2F)cc1 28996,c1(C(=O)NCCC(=C)CNC(=O)CCn2ccnn2)c(Br)cnn1C 28997,C(N=c1nc2scnc2c(N2CCOCC(F)(F)C2)[nH]1)c1n(C)nnc1 28998,C1(C(=O)N(C)CC2(C)CCCO2)(NC(C(CO)OC)=O)CCCCC1 28999,c1(C(=O)NCCN(C(Cc2c(SC)cccc2)=O)C)c(C)nn(C)c1-n1cncn1 29000,c1(C(N2C(C)CC(CNC(=O)CC3CCOCC3)C2)=O)cncc(C#N)c1 29001,c1(C(N2CCC(NC(C(CCC)OCC)=O)C2(C)C)=O)cc(F)cc(Cl)c1N 29002,c1(C(=O)NCC2(F)CN(C(=O)C=C3CCC3)C2)cc2cccc(Br)n2c1 29003,c1(C(=O)NCC(CC)NC(=O)CCc2scnc2C)cccc(C#CC2CC2)c1 29004,C(c1nc2cc(Br)cnc2s1)=C(C)C 29005,CC1(CNC(c2ccc(CNC(c3cccc(F)c3F)=O)o2)=O)CCCCC1O 29006,c1(CC(=O)NCCC2CCC(NC(C(C(=C)Cl)(C)C)=O)C2)ccccc1[N+](=O)[O-] 29007,C(=O)(C1=C(Cl)CCOC1)N1CCC(C(N2CC(CC)NC(=O)C2)=O)C1 29008,C(CN=c1nc(N2CC=C(Br)CC2)c2c([nH]1)CCS2)N1CC(C)OC(C)C1 29009,N1(C(CNC(CNC(CC(C)SC)=O)=O)=O)CCCC2OCCC12 29010,c1(CC)cn2c(n1)CC(C(=O)NCC(C)N(C)C(c1cc(C)cc(O)c1)=O)CC2 29011,N1(C(C(C)Oc2ccccc2)=O)CC2CC2(NC(C2(c3ccn(C)n3)CC2)=O)C1 29012,c1(CC)ccc(F)c(C(N2CC3CCOC3(CNC(=O)C(CC)SC)C2)=O)c1F 29013,n1(CC(N2C(C(=O)NCC(C)OC)CCC2)=O)ccc2ccccc12 29014,C1(C(N2CCCC2CCNC(C2(CF)CC2)=O)=O)CC12CCC(F)(F)CC2 29015,CCCCC(C)CCC(=O)N1CCC1CNC(c1sccc1CC#N)=O 29016,C(=O)(C1=C(C)OCCS1)N1CC(OCC)C(CNC(C2CCC(C)(C)OC2)=O)C1 29017,N1(C(C2(C)C(C)C2)=O)CC2CN(C(c3ccc(C(N)=O)cc3)=O)CC2C1 29018,N1(C(C2=CC(C)(CC)C2)=O)CC2CC(C1)CN(C(c1cc(Br)c[nH]1)=O)C2 29019,c1(OCC)ccc(C(=O)NCCN(C(=O)C2CC2)C2CC2)c(Cl)c1 29020,N#CC1CCN(C(=O)CC2CN(C(=O)CC3CCCOCC3)CC23CC3)CC1 29021,c1(CNC(c2n(CC(=C)C)nnn2)c2nc(CO)cs2)ccc2ccn(C)c2c1 29022,c1(-c2cn(CC(CNC(=O)C(C)(C)OC)OC)nn2)ccnc(NC(C)=O)c1F 29023,C(=O)(C1=CCOCC1)NC(COC)C(=O)NCCC1CCN(C)C1=O 29024,CN1N=C(C(=O)Nc2cccnc2C(N2CCCC(NC(N)=O)C2)=O)CCC1=O 29025,c1(C(=O)NCCC2CSCCN2C(=O)C=CCO)csc2c(F)cccc12 29026,c1(CCCC)ccc(C(N2CCN(C(C)C(=O)NC3(C(N)=O)CC3)CC2)=O)cc1 29027,c1(OC)nc(C)ccc1C(=O)NCC1(C)CN(C(c2c[nH]nc2C)=O)CCO1 29028,c1(C(N2CC(CC)N(C(=O)CCC(=O)OC)CC2)=O)cc2c(C)nn(C)c2s1 29029,c1(SCCC)cccc(C(=O)N(CC(C)(C)NC(C2CCOC2=O)=O)C)c1 29030,CC1CC2CN(C(=O)C(CO)C(F)(F)F)CC2N1C(=O)CCC(=O)C1CC1 29031,c1(CC)cc(C(N2CC(C(F)(F)F)(C(C)(C)O)C2)=O)no1.C12CC1(C)CNC2=O 29032,Cc1noc(C)c1C(C)C(=O)NCC1(CNC(C2(C)CNC(=O)C2)=O)CC1 29033,n1(CC)nc(C(N2CCN(C(c3c(OC)noc3C)=O)CC2)=O)c(Br)n1 29034,c1(C(N2CC(n3cc(C(C)(C)CO)nn3)C(O)C2)=O)cc2c(cn1)OCCC2 29035,Cc1cc(C)n(C(C)CC(=O)NCC2CCN(CC3CC(C)(C)CO3)C2)n1 29036,c1(OC)cc(C(=O)N(C2CC(NC(=O)C(CC(C)C)OC)C2)C)cnc1OC 29037,c1(C(=O)NCCC2(CNC(C(C)OCC=C)=O)CC2)scnc1C(F)(F)F 29038,CCCC(C)(C)CC(=O)NC1C(C)(C)C(NC(C2CSCCS2)=O)C1(C)C 29039,Cn1cccc(C(=O)NCC2C3CN(C(C4(CCF)CC4)=O)CC23)c1=O 29040,C1(NC(CSS(C)(=O)=O)=O)CCN(C(=O)CCN2CCCC2=O)CC1CO 29041,c1(NC(C2C3(CN(C(C)=O)C3)C2)=O)nc(Cl)ccc1I.c12ncc(o1)c(=O)[nH]2 29042,C1(NC(C)=O)CN(C(=O)C(Cc2cccc(Cl)c2)NC=O)CC2(CCOCC2)C1 29043,C1(C2CCN(C(=O)CC3OC(C)(C)OC3=O)CC2)(NC(C2CC(SC)C2)=O)CC1 29044,C12(NC(Cn3c(C(C)C)ncc3)=O)CCN(C(=O)COCCN(C)C)CCC1C2 29045,c1(C(=O)NC2CCC(CNC(=O)CCn3cccc3)C2)cc2c(=O)[nH]ccn2n1 29046,N1(C(CCN(C(=O)CCCCSC)CC=C)=O)CCCOC(C(C)C)C1 29047,C1(C(=O)NCCCC2(NC(=O)C=CCO)CC2)COc2c(F)cc(F)cc2C1 29048,c1(CNC(C(COC)C)=O)ccccc1CNC(C)=O 29049,C(C(C(=O)N1OC2CCC1C2)N(C(=O)C(Cl)Cl)CC)SCC 29050,C1(CC)CCN(C(c2ccc(O)cc2)=O)C1C(=O)Nc1cnsc1 29051,N1(C(C)=O)CCCC1(C)C(=O)NCC1C=CCN1C(=O)C=CCN1CCOCC1 29052,C1(NC(COCC=C)=O)CCN(C(c2ccc(OC)cc2N)=O)CC1F 29053,c1(C(=O)NCC(=C2CN(C(c3nc(OCC)oc3)=O)C2)F)cccc(C(C)C)c1 29054,C(=O)(CCC(=O)NCCC1(O)CN(C(c2cc(C(C)C)on2)=O)C1)NCC 29055,Cc1[nH]nc(C(=O)NCC(C)(C)CNC(=O)C(C)C(C)(F)F)c1[N+](=O)[O-] 29056,c1(C(C)=O)cccc(-c2cc(-c3nccn3CC3(C)CCCCC3)n[nH]2)c1 29057,c1(C(=O)NCC2(O)CCN(C(C3(CC4CC4)CC3)=O)C2)csc2ccc(F)cc12 29058,C1(NC(C(C)SCC)=O)CC(C(=O)N2CC=CC2(C)CO)=CC1O 29059,c1(C(N2CC(OC)C(NC(=O)C=Cc3cnc[nH]3)C2)=O)sc([N+](=O)[O-])cc1Cl 29060,CC1CCN(C(=O)C=Cc2ccccc2)CC1NC(=O)CC1CC(=O)NC1=O 29061,C1(NC(c2c(CC)ocn2)=O)C(C)CN(C(=O)C2=C(C)CCCC2)CC1C 29062,C1(NC(CSCC(C)C)=O)CCN(CCNC(=O)CC2CCS(=O)(=O)C2)CC1 29063,N1(C(=O)Nc2c(C(=O)OC)ccs2)CCN(C(c2cnccc2C)=O)CC1C#N 29064,c1(C(N2C(CNC(CC=CC)=O)CC(F)C2)=O)ccc(C)c(OC)c1F 29065,C1(C(N(CC(C)NC(c2cnc(O)s2)=O)CC)=O)CCC(NC(C)=O)CC1 29066,c1(CC)ncc(C(=O)NC(C)C(C)(C)NC(C2CC(n3ccnn3)C2)=O)s1 29067,CCCCC(O)C(=O)NCC(CC1CC1)C(=O)NC12CC1CN(C)C2 29068,C1(NC(CC(C)C)=O)CCCCCN(C(C23CC(CC(F)F)(C2)C3)=O)C1 29069,c1(C(=O)NCCCCC(C)NC(C(CC)OCC)=O)ccc([N+](=O)[O-])cc1C 29070,c1(C(=O)NCCNC(c2occ(C)c2)=O)ccccc1Oc1ccccc1F 29071,C(CC(C(=O)NC(C(C)(C)O)C1CC1)NC(=O)CCc1ccc(C)o1)=CC 29072,N1(C(c2c(OC)n[nH]c2)=O)CCC(CF)(NC(C2CSCCS2)=O)C1 29073,Cc1sc(-c2ccccc2)nc1C(=O)NC1CN(C(C2CCCO2)=O)C1 29074,C1(C(=O)NCC#CCNC(c2c(C)occ2)=O)C2CCC1(c1ccco1)C2 29075,C1(CC)CN(C)C(=O)CN1C(=O)NC1CCCC=C1Br 29076,N1(C(c2cncc(NC(c3ccncc3Cl)=O)c2)=O)C2COCC1CC(F)C2 29077,C(=O)(C1COc2ccccc21)NCC1CC(C)N(C(c2cc(F)ccc2N)=O)C1 29078,C1(C=O)CCCC(=O)C1.C1(COC)(NC(=O)CC2(N(C)NC)CC2)CCOC1 29079,C1(NC(c2cc(C)oc2)=O)CCCCN(C(c2c[nH]c(=N)s2)=O)CC1 29080,CCCCC(=O)C(=O)N(CCCNC(c1nnc(S)n1C)=O)Cc1cccnc1 29081,C=CC(F)(F)C(=O)N(CCCNC(=O)CC1COC(C)(C)C1)C 29082,c1(N2C(C3CCCN(C(C4CC(=C)C4)=O)C3)CCC2)nc2c(C)cccc2o1 29083,C12(NC(=O)C=CCO)CC(CO)(C1)OC21CN(C(=O)C2CCCc3ncnn32)C1 29084,C1(CC(=O)N(CCNC(C(N(C)C)C2CC2)=O)C2CC2)OCCCO1 29085,c1(NC(CN(C(C2N(CC#C)CCC2)=O)C)(C)C)nc2cc(Cl)cc(Cl)c2o1 29086,c1(N2CCN(C(=O)OC)CC2)nc(=N)[nH]c(=NCC(C2CC2)C2CC2)[nH]1 29087,c1(CC)nc(Cl)nc(N2CCCCC(CNC(C3(CO)CCCO3)=O)C2)c1C#N 29088,C12(C(=O)NCC3CCN(C(C(=O)NCC)=O)C3)C=CC(CC1)C2 29089,C1(NC(C2CC(C#C)(O)C2)=O)CCCC(C(=O)N(C)Cc2occc2C)CC1 29090,CC(C)(F)CC(=O)NC1(CF)CCN(C(=O)CCNC(=O)OC(C)(C)C)C1 29091,CC1(C)CCCC1(O)CNC(=O)CC1(NC(C2OC3CCC2C3)=O)CC1 29092,CCCCC(O)CCC(=O)NC1CCSC12CN(C(=O)Cc1ccc(F)cc1)C2 29093,Cc1noc(Cl)c1CC(=O)NC1(C)CCN(C(=O)CCCn2cnc(C#N)n2)C1 29094,c1(C(N2C(C)CC(NC(c3nccn3C)=O)C2)=O)ccccc1S(=O)(=O)C(F)F 29095,C1(NC(C2N(C(C)C)C(=O)CC2)=O)CCCCN(C(=O)C(F)C2CCC2)C1 29096,Cc1cccc(C(=O)NC(C)CN(C)C(C2(C)CCN(C)C2=O)=O)c1C#N 29097,CCCC(CCCNC(=O)Cc1ccc(Br)cn1)NC(c1c[nH]ccc1=O)=O 29098,CC1(C(=O)N(CC(N2CC(c3cc[nH]n3)C2)=O)C2CC2)COCCO1 29099,C(=O)(C1=C(Cl)CCC1)NC(CCCCNC(C(CC)(C)C)=O)C 29100,n1(CC)nccc1C=CC(=O)NCCCCNC(C1CCCC(C(F)(F)F)O1)=O 29101,CC(CC(=O)N1CCC(c2ncco2)C1)C(C)(C)NC(=O)CCc1ccncn1 29102,C1(CNC(C2(OC)CCSC2)=O)CN(C(c2c[nH]c(=O)cn2)=O)CCC1(F)F 29103,CC1CC=C(C(=O)NCc2cncc(C(=O)NCc3ncccc3F)c2)CC1 29104,C(=O)(CC(C)(C)C(=O)N(CCCN(C(=O)C(=Cc1cccnc1)C)C)C)OCC 29105,C(CCCCC(=O)NC1CC(NC(=O)CC2CC(F)C2)C12CCC2)OCC 29106,c1(C(C)=O)ccc(CC(=O)NC2CC(C)(NC(C3(C4CCCO4)CC3)=O)C2)cc1 29107,N1(C(C(CCCC)NC(N)=O)=O)CCC2(C1)CN(C(C1CSC1)=O)C2 29108,c1(N(C)C)cc(F)c(NC(C2CCN(c3ccc(Cl)cc3)C2=O)=O)cc1[N+](=O)[O-] 29109,c12cccc(Cl)c1OC2.c1(CNC(=O)NCCCOCC)ccc(F)cn1 29110,C1(CCC(=O)NC2(CNC(C(C#N)C3CC3)=O)CC2)NC(=O)NC1=O 29111,C1(CCC)(C(N2CC(O)(C(F)C(=O)N(C)C(C)C)C2)=O)CC(=O)C1 29112,N1(C(c2n[nH]cc2Br)=O)CC(NC(c2ccc(C3CC3)o2)=O)C2(CC2)C1 29113,c1(C(=O)NCCN(C(c2cnn(C(F)F)c2)=O)CC)cc(N)c(Cl)c(O)n1 29114,C(CN=C(NC1CCC1(C)C)N1CCCC2(CC2)C1)N(CC)CC 29115,c1(C(=O)NCC2CCN(C(C(OC)OC)=O)CC2C)cc2c(C)ccc(F)c2o1 29116,C(c1ccco1)=C(C)C(N1CCC(CNC(=O)C(F)=C2CCCC2)C1)=O 29117,CCC(C)(O)C(=O)N1CC(C(C)NC(C2(O)CCC2)=O)C1 29118,N1(C(C2=NOC(C)C2)=O)CC(C)(C)OCC1CNC(C12CCC(C)(CC1)OC2)=O 29119,C1(C)(C(=O)Nc2cc(C)sc2)CCCN1C(c1ccc(C(N)=O)[nH]1)=O 29120,C#Cc1ccc(CNC(=O)C(CC2CCOCC2)NC(=O)C(CC)OC)cc1 29121,C1(NC(=O)COCc2cscn2)CC2CCC(C1)N2C(=O)CCOCC(F)F 29122,CC1CN(C(=O)C=Cc2cncc(F)c2)CC1(C)CNC(c1ncncc1F)=O 29123,N1(C(CCCC)=O)CCCC2(C1)CN(C(c1cc3ccc(C)cn3n1)=O)CCO2 29124,Cc1cc(C(=O)N(CCNC(c2ccn(CC#N)n2)=O)CCOCCO)sc1C 29125,CC1(C)CC2(CC(C(N3CCC(CNC(=O)CCS(N)(=O)=O)C3(C)C)=O)C2)C1 29126,CCCCC(O)CC(=O)N1CC2C(C(=O)N(CC(=O)N(C)C)C(C)C)C2C1 29127,N1(C(c2ccc(COC)o2)=O)CCCCC(CNC(=O)C(CBr)=CC2CC2)C1 29128,c1(C(=O)NCC(CC(C)C)NC(C2NC(=O)C3CC23)=O)cn2c(n1)CCC2 29129,C(=O)(C(C)C(F)(F)F)NCC1C(CNC(Cn2c(CCC)nnc2S)=O)C1 29130,C1(C(N2CCC(CNC(C3CC4CCC3CC4)=O)C2)=O)CCC2CCC1O2 29131,C(c1cccc([N+](=O)[O-])c1)=CC(N1CC(C)C(NC(=O)COC(F)F)C1)=O 29132,c1(OC)ccc(NC(C2CCCN2C(C2CCC2)=O)=O)cn1 29133,Cc1c(CC(N2CCCCC2c2cn(-c3cccc(N)c3)nn2)=O)nc(Br)n1C 29134,C#CC1(O)CC(C(=O)NC(c2cnn(C)c2)C(=O)NC2CC(C)(CO)C2)C1 29135,c1(CC(=O)NC2CN(C(CC(C)C)=O)CC2C)c[nH]c2c(Br)cccc12 29136,Cn1nc(C(=O)NC2CCN(C(C34CC(C)(C3)C4)=O)C2)cc1Br 29137,C1(CNC(C2(Cc3ccccc3Cl)CCOCC2)=O)NCC12CCC2 29138,N1(C(C2C(C=C)C2)=O)CCC(NC(=O)Cc2sc(O)nc2O)CC1c1ccccc1 29139,c1(SC)ccc(C(N2CC(C)(NC(C3CC4CC4C3)=O)C2)=O)cc1Br 29140,c1(C(=O)NCCOC2CN(C(C(CCCC)O)=O)C2)ccc(Cl)c(S(N)(=O)=O)c1 29141,n1(CC(=O)NC2C(CNC(c3c(CC)cco3)=O)C2)c(C)nc2ccccc12 29142,c1(CC)ccccc1CC(N1CC(CNC(=O)C=C(C)c2ccco2)(OC)C1)=O 29143,Cc1nccc(C(=O)NC2(C(=O)NCC#CC3CC3)CCN(C)C2)c1N 29144,C1(O)(CC)CCN(C(c2ncccc2OCC(F)(F)F)=O)C1 29145,c1(C(N2CC3CCN(C(CC(C)C(F)(F)F)=O)C3C2)=O)cnn(C)c1S(N)(=O)=O 29146,C1(C(N2CSCC2C(N)=O)=O)(CC)CNC(=O)C1 29147,C1(C)(CC)CC(C(=O)NCC(CO)NC(=O)CC2CSCCO2)C1 29148,N1(c2nc(=NCCS(C)(=O)=O)[nH]cc2)CCOCC12CCS(=O)(=O)C2 29149,N1(C(C(N2CC(C(C)NC(C(CCC)C)=O)C2)=O)C)C(=O)NC2(CCCC2)C1=O 29150,C1(NC(c2n(C=C)ncc2)=O)CC2CC1CN(C(=O)CCc1cccnc1Cl)C2 29151,N1(C(c2c(COC)ccs2)=O)CCN(C)C(CNC(c2ncc(C)cn2)=O)C1 29152,O=S(=O)(c1cc2sc(=NCCCCO)[nH]c2cc1Cl)NC1C2CCC(F)(F)C12 29153,N1(C(c2ccon2)=O)CCC(Cc2cn(C3CCCC3O)nn2)CC1 29154,Cc1cc(NNC(=O)C2CCCN2C(c2cccc(C(C)C)c2)=O)cc(C)c1Br 29155,c1(C(C)OC(=O)C(C)Sc2ccccc2)cccc(OC(F)(F)F)c1 29156,C1(C(=O)NC(C(CC)C)CO)CCN(C(=O)C2=CCCCC2)CC1C 29157,C(=O)(C(CC(C)C)NC(=O)OC)NC1CCN(C(CNS(CC)(=O)=O)=O)C1 29158,CC1=C(C(=O)N2CC(NC(c3cc(Cl)cn3C)=O)CC2CO)CCCC1 29159,c1(N2CCC(NC(=O)NCc3cc(Cl)ncc3Cl)CC2)ncc2c(n1)CCC2 29160,c1(C(N(CCC)CCNC(=O)CN(C)C(N)=O)=O)cc(F)ccc1OC 29161,O=C(CCCCN1CCCC1)NCC12CC1CN(C(C1(O)CCSC1)=O)C2 29162,Cc1c(C(=O)NCC2CCN(C(C3CCOC3)=O)C2(C)C)c(Cl)nn1C 29163,c1(CCC(=O)NC(C(C)C)CNC(C2(C(C)(F)F)CC2)=O)ccc(F)cc1F 29164,Cc1ccn(C)c1C(=O)NCCC1CN(C(C2CC2C(C)(F)F)=O)CCO1 29165,C1(C)(CNC(C(CCC)C)=O)COCCN(C(c2ccc(CO)cc2F)=O)C1 29166,c1(OCCCC)sc2ncn(-n3cc(-c4ccccc4F)nn3)c(=O)c2c1C 29167,c1(OC)ncnc(C(=O)NCC2(O)CN(C(=O)Cc3ccc(C#N)cc3)C2)c1F 29168,N1(C(CCC=C=C)=O)CCN(C(=O)C(C)(C)COC)CC1C(C)C 29169,c1(C(=O)NC2CC(CNC(Cc3nc(C)sc3)=O)C2(C)C)ccc(CO)c(Cl)c1 29170,Clc1ccc2c(c1Br)CN(c1ccn3nccc3n1)CC2 29171,O=C1CCCC2C(C(N3CCCC3c3ccsc3)=O)C12 29172,CN1CCC(C(N2CCCC(Cc3cn(CSC4CNC(=O)CO4)nn3)C2)=O)CC1 29173,c1(C(N(C)C(C2(N(C)C)CCCC2)=O)=O)ccc(C23CCC(C2)OC3)cc1 29174,Cc1nc(S)sc1CC(N1CCC(F)(CNC(c2cncc(F)c2)=O)C1)=O 29175,C1(N(C)CC)CN(C(c2ccc(C3CCC3)cn2)C(=O)NC)CC12CCC2 29176,C1(NC(c2cc(CN(C)C)on2)=O)CCCCC1CNC(=O)C(C)(C)C1CCC1 29177,Cn1ccc2cc(-c3nc(-c4ccncc4)nn3CCc3ccccn3)ccc12 29178,c1(CN(Cc2occc2C)CCOC)scc2c1CCCC2 29179,c1(C(N2C(C)CC(NC(C(CCC)(C)O)=O)C2)=O)c(F)cc(F)cc1F 29180,c1(CC(=O)N(CC(C)O)CCNC(CCc2cnc(C)s2)=O)ccccc1C 29181,C1(CCC2N(C(c3ccsc3OC)=O)CCC2)CCCCN1C(c1ccoc1)=O 29182,N1(C(c2c(CC)c[nH]c2)=O)CCOC(CNC(=O)C(C)(CO)OC)C1 29183,CCCCC(C)(F)C(=O)N(CC(C)NC(c1cc(N(C)C)ccn1)=O)C 29184,N1(C(CC(C)(C)NC(=O)CC2CC3C=CC2C3)=O)CCC2C(C1)C2(F)F 29185,C1(C(=O)NCC(C)NC(C2CC3CCC2O3)=O)CCCCN1C(=O)OC(C)(C)C 29186,N1(C2CCN(C(=O)CCF)CC2)C2CCC1CN(C(C1C=CCC1)=O)C2 29187,C(C(F)(F)C(=O)NC1CCC1CNC(c1cnn(-c2ccccc2F)c1)=O)OC 29188,c1(C(N2CCC(CNC(C3(C)CC3(F)F)=O)C2)=O)cc2nc(F)ccc2o1 29189,C=CCCC(c1nnnn1CCCSC)NC(C)CNc1cnc(SCC)s1 29190,O(C1CCCc2ccccc21)C(C(C)OC(=O)CS(=O)(=O)c1cnn(C)c1)=O 29191,C=C(Cl)CCC(=O)NC(c1ccccc1)CNC(c1cnccc1Br)=O 29192,C(=O)(C1=C(Cl)CCC1)N1C(CCNC(CSCC)=O)CCC1 29193,N1(C(c2ccc(CC)cc2)=O)CC2CCC1CN2C(=O)C(c1csc(C)n1)=O 29194,c1(CC(=O)NC2(CO)C(C)C2)csc(-c2cccnc2)n1 29195,C1(CC(=O)NC(C2CCN(C(=O)C(F)CC3CCOC3)CC2)(C)C)SC(=N)NC1=O 29196,C1(NC(c2c(SC)cn(C)n2)=O)C2COCC1CN(C(C1CCCO1)=O)C2 29197,c1(C(=O)NC23CCN(C(Cc4c(C)ocn4)=O)CC2C3)ccc2c(c1O)CCC2 29198,C1(CCCNC(c2cnsn2)=O)CCCCN1C(=O)CCC1CC1 29199,CC(C)C(C(=O)NC1CC(CNC(c2nocc2Cl)=O)C1)N(C)C 29200,n1(CC)nc(C)cc1C(=O)N(C)CC1CCCC1NC(C1(C)CC1C)=O 29201,c1(CCC(=O)NCC(C)NC(CCOC)=O)ccc(Br)cc1 29202,c1(C(N2CC(NC(CC(c3ccccc3F)C)=O)C2)=O)cc2c(s1)CCCCC2 29203,c1(-c2cn(C(C(=O)NCc3ncc(C)o3)C)nn2)cc(Cl)c(Cl)c(Cl)c1 29204,C1(N2CCC(C(=O)Nc3c(C)n(CC(F)(F)F)nc3)C2)CCN(C)CC1C 29205,c1(C(=O)NCC(F)CNC(C2(CO)CC2)=O)cc2sc(Br)cc2[nH]1 29206,Cn1c(C(=O)N(CCNC(C2CC2F)=O)CC2CC2)cc2occc12 29207,Cc1nc(O)[nH]c1C(=O)N(C)CC1(O)CCN(C(=O)C(C)Cc2ccnn2C)C1 29208,N1(C(C(C)OCCOC)=O)CC2CC(C(N3CC(C(F)(F)F)C3)=O)(C2)C1 29209,C1(C(N2CCN(C(=O)Cc3cccnc3)CC2)=O)CC12CCCOC2 29210,c1(CC(N2CCC(C(=O)OC)CC2(C)C)=O)cccc2c1CCCC2 29211,C(c1ccc(Cl)cc1F)=CC(=O)NC1CCC(CNC(c2n(CC)ncn2)=O)C1 29212,C(C)(CCC(=O)NCC(c1ccc(OC)cc1)NC(=O)CCOC)OC 29213,c1(C(N(CC(CC)NC(C2CC23CCOCC3)=O)C)=O)ccc(C)c(C2CC2)c1 29214,c1(C(=O)OC)ccc(CCc2cn(-c3ccc(C(=O)NO)cc3)nn2)cc1 29215,c1(C(=O)NCCN(C)C(c2nocc2Cl)=O)cncc2c1CCC2 29216,c1(NC(COc2ccc(C)cc2)C)cc(=NCCS(N)(=O)=O)[nH]c(C)n1 29217,c1(C(N2CC(C(C)NC(CC(COC)C)=O)C2)=O)ccc2c(c1)CCO2 29218,N1(CCC(=O)NC(C2CCCN(C(=O)CCF)C2)C)CCCCC1=O 29219,c1(OC)ccc(C(=O)NCCCCCCNC(C2CCCCN2C)=O)nc1N 29220,Cc1cccc2oc(C(=O)NC3CC(O)C3(C)C)cc12 29221,C1(OC)COc2c(C(=O)NC34CC5CCC(C3C4)N5C(=O)CSC)cnn2C1 29222,Cc1nccn1CC(=O)NC1(C(=O)NCCN2CCC(C)C2)CCC1 29223,N1(C(c2ccno2)=O)CC(N=c2cc(C3CC3)nc(Cl)[nH]2)C2(CCOCC2)C1 29224,C1(NC(C2(NC(CSCCCC)=O)CCC(C)(C)C2)=O)CC(C2CCCC2)C1 29225,CC1(NC(c2cc(C3CC3)n[nH]2)=O)CCCN(C(=O)C(F)F)C1 29226,N(C1CN(C(=O)Cc2ccoc2)Cc2ccccc21)c1nc(C)nc(O)c1C 29227,CC1(C)CCC2CC(NC3CCCOC3)c3cccc1c32 29228,c1(NC(C=CC(C)(C)NC(C2CCC3(CC3)C2)=O)=O)cnc(F)nc1 29229,N1(C(C(C)=C2CC2)=O)CCCC2CN(C(=O)Cc3cncc(C#N)c3)CCC12 29230,c1(CN(C(c2ncc(Cl)n2C)C(=O)NCCCC)C)noc2ccccc12 29231,C(C(=O)NCCn1cc(CSCCO)nn1)(C(C)(C)O)NC(=O)OC(C)(C)C 29232,c1(CC(=O)NC(CN(CC)CC)C)cccnc1.C(C(C)(C)CO)N 29233,c1(CN2C(C(=O)NCc3nc(C(F)(F)F)cs3)CC2)csc2ccccc12 29234,Cc1cnn(C)c1C(=O)NC1CCC(CNC(c2ccc(NC(N)=O)cc2)=O)C1 29235,c1(C(N2C(C(=O)NCCc3c(C)nn(C)c3)CC2)=O)cc(C#N)cn1C 29236,Cc1ccc2c(c1)CC(C(N1CCCC1CCCNC(c1cc(C)no1)=O)=O)S2 29237,C12(C(=O)NC(c3cnc[nH]3)C)CCCC1CCN2C(C1OCCO1)=O 29238,C=CCCCC(=O)NCCC1(NC(=O)C(C)NC(C2CCCC2)=O)CCCC1 29239,C1(NC(CC2CCCC(CC)C2)=O)CC12CCN(C(c1ccc[nH]1)=O)CC2 29240,C=Cc1ccc(C(N2CCCC2CC(=O)NCCc2ccc(Cl)cc2)=O)cc1 29241,CCCCN=C(NCc1ccnn1C)NC1CCN(C(c2ccncc2)=O)C1 29242,c1(C(=O)NCCCCC2CCCN(C(=O)CO)C2)cc(Cl)c2c(c1)OCCCO2 29243,CC(C)CC(CNC(=O)CSCC(C)C)NC(=O)CSc1cccs1 29244,c1(C(c2nnn(C)n2)N(C)C(N2CCc3ncncc3C2)=O)cncc2ccccc12 29245,C#CCC(C(=O)NC1CCN(C(=O)C(C)O)C1)C1CC1 29246,c1(C(N(C2CC3CNC2C3)C(CC)CO)=O)ccc(C(N)=O)cc1 29247,N1(C(C=Cc2cn(C)nn2)=O)C2CCC(C2)C1C(=O)NCc1ncn(C)n1 29248,c1(NC(C(COC)(C)C)c2nnnn2CCSC)ccc2nsnc2c1 29249,N1(C(CC2C(C)=NNC2=O)=O)CC2CCC1C1CN(C(c3cnc(C)o3)=O)CC21 29250,N1(C(C(=O)OC)C)CCC(C(N2CCCCC2CO)=O)(OC)CC1 29251,C1(C(=O)NCCOC2CCN(C(CC3CN(C)CC3O)=O)C2)CCCCCCC1 29252,C=C=CC(C)C(=O)N1CC(O)(CCNC(=O)CCOC2CCOC2)C1 29253,c1(C(=O)NCC(=C)CCNc2cc(=O)n(C)cn2)ccc2c(c1)COCC2 29254,N1(C(c2cnn(C)n2)=O)CCC(C(N2CCCC(CC3CC3)C2)=O)C12CCC2 29255,CCS(=O)(=O)c1ccc(F)c(C(=O)NC(C)C(C)NC(=O)Cc2cccs2)c1 29256,C12(NC(CC(C)O)=O)CCC(CC1)N(C(=O)Cn1cnc([N+](=O)[O-])n1)C2 29257,C#CCC(C)(C(=O)NC1CC(COC)C1)NC(C1CC(=O)CS1)=O 29258,C1(NC(CC(COC)NC(C2CC3(C2)CC32CC2)=O)=O)CCCCCC1(C)C 29259,C(C(C)(O)CCC)NC(C=C(CNC(C(C)OCC#C)=O)C)=O 29260,N1(C(C2C(OC)CC2)=O)CC2C(C(=O)N(C)CC3CCCS3)C2C1 29261,c1(C(N2CCC(C)(CSC)C2)C(=O)NC2CCCC2)cc(SC(C)C)cc(C)c1 29262,N1(C(C2C(C)C2)=O)CCCC1CN(C(=O)CCc1nc(-c2ccsc2)no1)C 29263,c1(C(N2C(C)(CNC(=O)CS(C)(=O)=O)CCC2)=O)cc(=O)n2ccccc2n1 29264,N1(C(c2cnc(C(C)OC)s2)=O)CCCC(N(C)C(c2c(C)nsc2C)=O)CC1 29265,N1(C(c2ccc(CC)cc2O)=O)CC2CC(NC(c3snc(Cl)c3Cl)=O)CC2C1 29266,N1(C(CC2CC(C)(C)OCC2)=O)CCC2(CCCN2C(=O)C(O)C2CCC2)C1 29267,c1(C(=O)NC2CN(S(C)(=O)=O)C2)cn2cc(-c3cncc(C4CC4)c3)ccc2n1 29268,S(=O)(=O)(c1c[nH]ccc1=NC1CC1C1CCCC1)NCc1scc(C(C)C)n1 29269,C=C(C)CC(C(=O)NCCCCNC(N)=O)NC(c1ccsc1)=O 29270,C1(C)(C(N2CCC(NC(c3ccn(C)c3)=O)C(CO)C2)=O)CC(C2CC2)=NO1 29271,Cc1cccc(Cn2cc(NC(C3(NS(C)(=O)=O)CC4CCC3C4)=O)cn2)c1I 29272,Cn1cc(-c2cc(C(=O)NC3(C)CN(C(C4(c5nccs5)CC4)=O)C3)no2)cn1 29273,C1(C#CC(=O)N2CCC(OCCNC(C3CC3F)=O)C2)(CC)COC1 29274,C1(C)(NC(C=CC)=O)CCN(C(c2oc(-c3ccccc3)nc2C)=O)C1 29275,C1(CNC(CC(CC)SC)=O)CCCCCN1C(=O)COc1cc(C)ccc1C 29276,n1(CC)nnc2c1CCC(C(=O)N(C(CNc1ncccc1C#N)C1CC1)C)C2 29277,N1(C(CNS(CCCC)(=O)=O)=O)CC2CCCN(C(=O)C(C)C(F)F)C2C1 29278,S(=O)(=O)(c1ccc(=NCc2ccc(S(C)=O)cc2)[nH]c1)N1CC(CC)N(C)CC1 29279,C1(OC(C(CCC)(C)C)=O)CCCN(C2CCCc3ccccc32)C1=O 29280,Cc1oc(C(=O)NCCNC(C2CCCCN2C2CCCC2)=O)cc1S(N)(=O)=O 29281,C(=O)(C(C(=O)NCC(C)(C(C)C)NC(=O)C1=CCC1)c1ccccc1)OCC 29282,C(=O)(CCC(C)(C)NC(c1cc[nH]c(=N)n1)=O)N(C)Cc1onc(CC)n1 29283,c1(CCNC(C2CCN(c3ncc(I)cn3)CC2O)=O)c[nH]c2ccc(Br)cc12 29284,c1(C(=O)NCC2CCCC(NC(CCCSC)=O)C2)coc2c(F)cc(Cl)cc12 29285,c1(C(N2CC(CNC(CN(S(C)(=O)=O)C)=O)C3C2C3)=O)cc(N)c(Cl)c(O)c1 29286,N1(C(C(c2cccc(O)c2)C)=O)CC(CNC(C2(C)COC2)=O)C(C)C1 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29357,c1(C(=O)NCCCN(C(CCC=CC)=O)CCO)cnc(N2CCOCC2)nc1 29358,c1(C(C)=O)cc(NC(C2CC2C(=O)Nc2ccc(Br)c(F)c2O)=O)cc(C#N)c1 29359,N1(C(CCC2(C#N)CCC2)=O)CCOCC(NC(C2CC3CCCCC23)=O)C1 29360,CC1(C)C2CN(C(C3CC3F)=O)C(C(N3CCCC(O)C3)=O)C12 29361,C#CC1(C(=O)N(C)CC2CN(C(=O)Cc3csc(C)n3)CCO2)CCOCC1 29362,CCCC(C)CC(C(=O)NC(C)(C)C)N1CCCC1(CC)CO 29363,C1(NC(CC(COC)C)=O)(CO)CCCN(C(=O)Cc2conc2C)C1 29364,c1(C(N(CCN2CCOCC2)CC)=O)cn(CCNC(=O)Cc2ccsn2)nn1 29365,N(C1CC(F)(F)c2cc(Br)ccc21)C(N1CCC(O)(c2ccccn2)C1)=O 29366,c1(-c2cn(CC3CCN(C(=O)Cc4ncccn4)C3)nn2)cccc2c1OCO2 29367,CCCC(CCNC(=O)CN(C(=O)CC1CCCN1C)C(C)C)C1CC1 29368,C1(CC)CCN(C(=O)CC(C)C2CC2)C1CNC(c1ccnc(C(F)F)c1)=O 29369,S(=O)(=O)(c1ccc(F)cc1)NCCC(=O)N1CC(CNC(C2CC(C)C2)=O)C1 29370,C1(C(N2C(C(C)NC(c3c(C)occ3)=O)CCC2)=O)CSC(c2ccccc2)=N1 29371,c1(CCNC(CN(C(C(c2cncnc2)C)=O)C2CC2)=O)ccnn1C 29372,c1(C(N2CCC(CCNC(C(C)=CC)=O)CC2C)=O)cccc2c1ccn2C 29373,C1(NC(Cc2ncc(CC)[nH]2)=O)CCCN(C(=O)CSCC2CCCCO2)C1 29374,n1(CC)ncc(C(=O)N(CCCNC(=O)COCP(C)(C)=O)C2CC2)c1Cl 29375,C1(CNC(C2C(C(=O)OC)C2)=O)CCCC(CNC(c2ccc(C)cc2)=O)C1 29376,C1(C(N2CCC(c3cn(-c4ccncc4)nn3)C2)=O)(SC)CC(=O)C1 29377,CC1CN(c2cc(NC3CC4OC(=O)CC34)ncn2)CCC1N(C)C 29378,c1(CC)ccc(C(=O)NCC2(C)CCCN(C(c3csnn3)=O)C2)c(O)c1 29379,C1(C(=O)NCC)(N(C(=O)COCCCOC)C)CCOC1 29380,N1(C(C2(O)CCN(c3c(OC)nccn3)C2)=O)CCOCC(O)C1 29381,C1(NC(C(CC2CCOCC2)NC(C2CCCO2)=O)=O)CC2CC1CC2CO 29382,O=S(=O)(c1cnc(NC2CC(CF)C2)c(Cl)c1)NC1CCC2(CC1)CC(O)C2 29383,Cc1c(NC(C2(F)CN(Cc3ccc(Br)s3)C2)=O)cccc1F 29384,c1(CN(C(c2snc(C)n2)C(=O)Nc2ccccc2)C)ccnc(Cl)c1 29385,c1(COC)ccc(CNC23CC(C(=O)NC(C)CC(=O)OC)(C2)C3)cc1 29386,N1(C(C(c2ccccc2F)C)=O)CCCC(CO)(NC(c2cccn2C)=O)C1 29387,CC(C)(O)C(F)C(=O)NCCC1CC(F)CN1C(=O)C1CC1 29388,C(C(C(C)(C)C)NC(=O)CCc1nc(C(C)OC)no1)NC(C1C(CC)C1)=O 29389,c1(CCC(=O)NC(C)CC(=O)N(C)C)ccc(Cl)nc1 29390,c1(N2CCN(C(C(=O)NC)C)CC2)nccc(=NC(C)c2ccn(C)n2)[nH]1 29391,N1(C(CSc2cccc(C(C)=O)c2F)=O)CCOc2c(F)cccc2C1 29392,c1(NC(C2CN(S(CC)(=O)=O)C2)=O)cc(-c2ccco2)nn1C 29393,CC1CCN(C(=O)CN2CCS(=O)CC2)CCN1C(=O)CC1CCCC(C)(C)C1 29394,C1(CNC(COC(C)C)=O)CCN(C(=O)C(C)(C)CC2CCOCC2)CC1C 29395,N1(C(C(C=C)(C)O)=O)CCc2nc(CNC(C3CC(C)CC(C)(C)C3)=O)sc2C1 29396,c1(CC)nn(C)cc1C(N1CCCC(NC(c2cc(C(=O)OC)c[nH]2)=O)C1)=O 29397,CCCCCC(C(=O)NC1CCCCC1)N1CCC2(CSC2)C1 29398,C(CN=c1ccc(C(=O)NCc2nc(CNC(=O)CCS(C)=O)cs2)c[nH]1)OC 29399,N1(C(C(CC)=CCCC)=O)CCN(C(=O)CCc2nncnc2O)C(CO)C1 29400,N1(C(=O)COC2CCCC2O)CC2CCCC(C1)N2C(C1CC(F)(F)C1)=O 29401,C(C(CC1CCCC1)C(=O)Nc1ccc(SC)cc1)NC(CC(=O)NCC#C)=O 29402,c1(C(=O)NC(CCCNC(C(Cn2ccc(C)n2)C)=O)(C)C)cnc(N)c(N)c1 29403,c1(C(=O)NC2CC(NC(CCC(=C)Br)=O)C2)ccnc2c1nnn2C 29404,CC(C)C(C(C)NC(c1csnn1)=O)NC(c1ccc(C(C)(C)C)nc1)=O 29405,C(C1c2ccccc2CCN1C(c1conc1C)=O)NC(C1(COC)CC1)=O 29406,N1(C(c2c(C)c(Br)n(C)n2)=O)CCCC(C2CN(C(=O)COC(C)C)C2)C1 29407,c1(NC(=O)NCCC2=CCCC2)ccc([N+](=O)[O-])cc1 29408,c1(CN2CCC3(C(C(=O)NCCc4ccc(F)nc4)C3)C2)cc(Cl)cc(Cl)c1O 29409,c1(C(CC=C(C)C)NC(=O)CC2CC(NC(=O)OC(C)(C)C)C2)cccnc1 29410,C1(CN(C(=O)Cc2cn(C)cn2)C)CCN(C(c2csc(C#N)c2)=O)CC1 29411,C(=O)(CCCCCNC(N)=O)NC(C)CCCCNC(C12CCC1C2)=O 29412,C1(CC)CC(C(=O)NCC(c2ccsc2)O)CCN1C(c1csc(C)n1)=O 29413,N1(C(CNC(C2C(C)CC2)=O)=O)CCSCC1C(N1CC(N(C)C)C1)=O 29414,N1(C(C(C)=C(C)C)=O)CCN(C(c2nn[nH]c2C(F)(F)F)=O)C2(CCC2)C1 29415,Cc1cc(C(=O)NCc2ocnc2C(=O)NC2CC3CCC2C3)c(C)o1 29416,C1(C(N2CC3CC(C2)C(=O)N3)=O)CCCCC(C)(C)C1.C1(COCC)(CC)CC1 29417,Cc1nn(C)c(Cl)c1C(=O)NC1CCCC(NC(c2cc(CF)on2)=O)CC1 29418,C1(NC(c2ccnc(C)n2)=O)CCCCCN(C(c2ccc(C3CC3)cc2)=O)C1 29419,c1(NCCNC(c2nc(C(F)(F)C(=O)O)cs2)=O)ccc(F)cc1 29420,c1(C(=O)NCC2N(C(C(CC=C)(F)F)=O)CC2)ccc(C)c(OC)c1F 29421,C1(C(=O)NCC2N(C(C(CC)N3CCCC3=O)=O)CC=C2)CC2(C1)CC(C)(C)C2 29422,C(=O)(C1=CCCN(C(C2CC2C(C)(C)C)=O)C1)NC1CN(C)CC1(F)F 29423,C1(NC(N(CC(O)COCc2ccccc2)C)=O)CC12CCCCCC2 29424,N1(c2nnc(-c3c(C)ocn3)n2CC2CCOC2)CC2CC1c1ccccc12 29425,C(C(CCC(F)(F)F)Nc1nccc(N2CCC(F)CC2)n1)OC 29426,C(=O)(C1=NOC(C)(C)C1)NCC1C(N(C)C)CN(C(CC2CCCN(C)C2)=O)C1 29427,C(CC(CC)C(=O)NCC1CN(C(c2cnn(C)n2)=O)CC1O)=CC 29428,C1(NCC(C)Cn2cccn2)CCCC1NC1CN(C(=O)OC(C)(C)C)C1 29429,C1(NC(C2(OC)CCN(C(CCC#C)=O)C2)=O)CCn2nccc2C1 29430,c1(N2CC(N(C)Cc3cnn4c3CCCC4)C2)ncnc2cc(I)sc12 29431,C(=O)(C1CCCc2nc[nH]c21)NC(C)(CNC(c1snc(O)c1Cl)=O)C1CC1 29432,CC(C)C(C(F)F)NC(C1CCN(c2cccc(C(F)(F)F)n2)CC1)=O 29433,c1(C(N2CCC(CC(C)NC(C3C(C=C)CC3)=O)CC2)=O)c(C)nn(CC)c1C 29434,N1(C(CC=CCC)=O)CCOC(CNC(c2sc(-c3ncccn3)nc2C)=O)C1 29435,C(=O)(C1=C(C#N)CCC1)N(C1CCCC(NC(=O)C=CC2CC2)C1)C 29436,CCC(CC)(C(=O)NCCC1CN(C(C2(COC)CC2)=O)CC(C)O1)OC 29437,C12(NC(C=Cc3cncc(C)c3)=O)CCCC1CN(C(c1cccc(O)n1)=O)C2 29438,CC1CN2CC(C)N1C2.C1(C)(n2cc(-c3cnccc3Cl)nn2)CCC(=O)N1C 29439,C(=O)(CN=c1cc[nH]cc1)NC1CC(NC(c2cc(CC)no2)=O)C12CCC2 29440,C(=O)(CCC(C)(C)C)N1CC(NC(C(CC)C)=O)C(C)C1 29441,C1(C(N2CC(O)(C(CNC(C(C=CC)O)=O)(C)C)C2)=O)COc2ccccc2O1 29442,c1(OC)cc(C(=O)NC2CCCCC2NC(c2ncccc2N)=O)cc(F)c1F 29443,Cc1nc(C)c(C(=O)NC(C2CCN(C(C3CCCC3C(C)C)=O)CC2)(C)C)[nH]1 29444,c1(C(N2CC(C)(CC(=O)NCc3cc(F)ccc3Cl)C2)=O)cc(F)ccc1C#N 29445,c1(CC(=O)NC2(CCNC(CCCSC)=O)CC2)ccc(O)c(F)c1 29446,C1(NC(C2(CC#C)CCCC2)=O)CC2CC1CN(C(c1ncc(C(N)=O)s1)=O)C2 29447,C1(C(N2CCC(O)(CC)C2)=O)Cc2nnsc2S1 29448,C12(CNC(c3cc(CC)nn3C)=O)CN(C(=O)C=CC3CC3)CC1CCO2 29449,C1(NC(C2CCOCC2)=O)CS(=O)(=O)C2CN(C(c3ncccc3Cl)=O)CC12 29450,C1(COCC)CCN(C(=O)CN(C(c2ccc(CC)o2)=O)CC)C1 29451,c1(NC(=O)NC(c2nc(C)sc2)Cc2cccc(Br)c2)cc(F)ccc1O 29452,C1(F)(CNC(=O)Cn2c(O)nnc2O)CCCN(C(C2C3CC4C(C3)C24)=O)C1 29453,N1(C(c2nn[nH]c2Cl)=O)CCN(C(=O)C=CBr)C2CCCCC2C1 29454,C1(CNC(COCCCCC)=O)CC(CO)CO1.C12CC(C1)CNC2=O 29455,O=CN1CCCN(C(=O)CC2CC=CCC2)CC1 29456,C#CC1(O)CCN(C(=O)C(CC=CC)NC(c2ncccc2Cl)=O)C1 29457,N1(c2nnc(-c3ccc(CO)o3)n2CC2CCSC2)CCc2nc(Cl)ccc2C1 29458,c1(C(N2CCC(NC(C(CCC)OC)=O)C2)=O)coc2cc(OC)ccc12 29459,Cc1occc1C(=O)NCC(O)CCNC(=O)CC1(O)CCOC1 29460,CN1C(=O)CCC1CC(N1CCCCC1CCNC(c1csc(Cl)n1)=O)=O 29461,c1(NC(CC2CCN(Cc3ccc(OCC)c(Cl)c3)C2)=O)cc(Br)c(Cl)cc1F 29462,O=C(C1=NN2CCCN=C2N1)NC1(C(c2ccc(F)cc2)=O)CCOC1 29463,C1(C)(CNC(C23CC(CC)(C2)C3)=O)CCN(C(=O)CCCCc2ccccc2)C1 29464,c1(C(N(C)CC2CCCN(C(C(C)S(C)(=O)=O)=O)C2)=O)ccc(S(C)(=O)=O)s1 29465,C1(C(=O)NC(c2ccc(F)cc2Cl)c2n(C)ccn2)CCN2CCOCC12 29466,C(=O)(C(CO)C(C)(C)C)NC(CNC(c1ccc(C#C)o1)=O)CC(C)C 29467,C1(CNC(c2c(CC)onc2)=O)CN(C)CCN1C(=O)CCc1ccn(C)c1 29468,N=c1[nH]c2cc(C(=O)NCC3C4CN(C(=O)CSc5nncs5)CC34)ccc2o1 29469,c12cc(Br)c(C(F)(F)F)cc1OC(=O)C(CC)NC2=O.c1(SCC)cccc(F)c1 29470,N1(C(CN(CCC(c2scc(C)c2)O)C)=O)CCC(C)C(CCc2nn[nH]n2)C1 29471,C1(CC(=O)N(CCCNC(C=C(C)CCc2ccccc2)=O)C)CCC2CC2C1 29472,c1(C(N2C(C(=O)Nc3cc(C(C)=O)sc3)CNCC2)=O)c(Br)c(C2CC2)nn1C 29473,c1(C(=O)NC2C(CNC(C(C)(C)c3ccc(Cl)s3)=O)CCC2)cc2n(n1)CCO2 29474,N1(CCNC(=O)CC(F)(F)F)C(=O)CCN(CC2CCCc3nc[nH]c32)C1=O 29475,O=S(=O)(c1cc(Br)c(F)cc1F)NCC1CCN(Cc2cc[nH]n2)C1 29476,C(=O)(C(C)CCCC(C)C)N1CC(CC)(NC(=O)CNC(=O)C(F)(F)F)C1 29477,CONC(=O)C(=O)NC1CN(C(=O)COCP(C)(C)=O)CC1C 29478,C(=O)(C(C)(C)CCCNC(=O)C1=COCCC1)N1CC(C)C(C)C1 29479,n1(CCC(N2C(C(N)=O)C3CCCC32)=O)c(S)nc2ccccc2c1=O 29480,Cc1cc(C(=O)NCCC(C)NC(c2c(C)ccnc2C)=O)c2c(c1)CCCN2 29481,CCC(CC(=O)N1CCOCC1CCNC(=O)C=Cc1nccs1)C(F)F 29482,CC(C)(C)C1=NOC(C(=O)NCC2CCN2C(=O)C=C2CCCCC2)C1 29483,C1(CCC)(NC(=O)CC2(OC)CN(C(C3(CSC)CC3)=O)C2)CCNC1=O 29484,C(CC(=O)NC1(CO)CC2CCCC12)(CC(C)C)NC(C(C)NC(=O)OC)=O 29485,N1(C(CCCC#C)=O)CC2CCCC2C1C(=O)NC(C)CC(=O)NC 29486,Cc1cc(OCC(F)(F)F)c[nH]c1=NCc1ccc2c[nH]nc2c1 29487,C1(COC)(NC(c2cc(C(F)F)nn2C)=O)CCN(C(C2(F)CCCC2)=O)C1 29488,c1(NC)ccc(C(=O)NCCCCC(C)NC(c2cccc(F)n2)=O)cc1 29489,C(C(F)(C(=O)NCC1CC2CCC(C1)C2)C(C)C)NC(CCC(CC)=O)=O 29490,C(CCC1CC1)(C(=O)NC1CC2C=CC1C2)NC(C(C1CCC1)OCC)=O 29491,c1(CC)cc(C(N2CCC(N(C(=O)CC3CCCC(O)C3)C)C2)=O)c(C)o1 29492,C(=O)(C1(C)CCn2c(C)nnc21)N1CC(O)(CNC(C(CC)O)=O)C1 29493,C(=O)(C1CCCn2ncnc21)N1C2CN(C(c3nccc(OC)c3C)=O)C(C2)C1 29494,c1(OC)cc(C)c(C(=O)NCC2CC(O)CN2C(C2CCC(=O)N2C)=O)c(C)c1 29495,N1(C(c2[nH]cc(CC)c2)=O)CCN(C(c2sc(C(C)(C)C)nc2C)=O)CC1C 29496,C1(C(N2C(CNC(c3c(N)ccc(C)c3)=O)CC(F)C2)=O)CCc2ccnn2C1 29497,C1(C(=O)NC(CCNC(c2nn(CC)c(O)c2)=O)C(C)C)CCc2nccn2C1 29498,Cc1nc(C2CC2)nc(C)c1C(N1CC(NC(C2CC(C)OC2=O)=O)C1)=O 29499,C(=O)(C(O)Cc1cnn(C)c1)NCCN(C(C(c1ccc(Cl)s1)C)=O)C1CC1 29500,N1(C(Cc2ccc(OCC)cc2)=O)CC(NC(=O)C(C)NC(N)=O)CC(F)(F)C1 29501,c1(CC(=O)NCC2(NC(C(CC#C)O)=O)CCCCC2)cccc2c(C)csc12 29502,N1(C(CCC)=O)CC(NC(=O)CCCN(C(C)C)CC)C2CC2C1.C1CCO1 29503,c1(CN(OC)C(=O)NCCS(=O)(=O)NC2CC2)ccc([N+](=O)[O-])cc1 29504,N1(C(c2cc(C)c(CO)cn2)=O)CCC2CCCN(C(=O)C3=COCCC3)C2C1 29505,c1(C(COC)N(C)C(c2nnsc2C)=O)ccc(Cl)cc1 29506,c1(OC)c(F)ccc(C(N2CC(NC(c3ccc(Cl)o3)=O)CC2C)=O)c1F 29507,CC(CCCNC(c1ncoc1C(C)(C)C)=O)NC(=O)CN1CCOCC1 29508,c1(C(=O)OCC)nc(C(N2CCC(O)(CNC(=O)CC(C)COC)C2)=O)c(C)s1 29509,O(NC(=O)CCc1ccc(OC)cc1)CC(CC)C 29510,C1(CC(C)C)CC1N=c1[nH]c(N2CCCC(c3cccnc3)C2)nc2c1CCC2 29511,NS(=O)(=O)C1CC(C(=O)NCc2cccc(CNC(C3CC3CF)=O)c2)C1 29512,c1(CC(=O)NC2C(NC(CCN(CCC)C)=O)CC2)csnc1C 29513,C#CCC(C(=O)NC)NC(C1CC(NC(=O)C(C)OCC2CC2)C(O)C1)=O 29514,C1(F)(CNC(C2(SC)CCC2)=O)CCN(C(c2coc(C3CCOCC3)n2)=O)C1 29515,c1(C(N(C)CCNC(=O)CCOC2CCC2)=O)c[nH]c2cccc(F)c12 29516,c1(NC(c2c(O)cn(-c3ccc(OC)cc3)n2)=O)c(Cl)cc(Br)cc1Cl 29517,c1(C(C)C(N2CCCC3CC23)=O)cc2ccccc2o1 29518,C(=O)(CC1=NN(C)C(=O)C1)N1CCC(C)CC1CNC(C1CNC(=O)O1)=O 29519,C(CC(C(C)(C)C)NC(c1cc(C2CC2)cs1)=O)N(C(=O)CCCN1CCCC1)C 29520,C1(N(C)C(C2CCNC2=O)=O)CN(C(c2cc(C(C)(C)C)ccn2)=O)CC1(C)C 29521,N1(C(c2c(OC)n[nH]c2)=O)CC(C)(C(=O)NCc2ncc[nH]2)CC1(C)C 29522,C1(NC(Cc2cc(COC)on2)=O)CN(C(=O)CP(C)(C)=O)CCC1C 29523,C(C(N=c1cc(C)nc(NC2CC3(C2)CC(O)C3)[nH]1)C1CC1)OC 29524,c1(NC(=O)CCC2(NS(=O)(=O)Cc3ccc(Br)cc3)CCC2)ccc(CO)cc1 29525,Cc1nc(Br)c(Cl)cc1NC(=O)NC(c1ccn(C(C)C)n1)C 29526,N1(C(C=C(C)CNC(C2(O)CCCC2)=O)=O)CCC2CCN(C)C2C1 29527,C1(C(N2CC(NC(CC=CC=C)=O)(CO)C2)=O)CCCC2(CCC2)O1 29528,C(=O)(CC(C)(C)CC(=O)NCC1CC1CNC(C1CC2(CCC2)C1)=O)OC 29529,C(CC(C)C)(C(=O)NCC(CNC(=O)CCc1cnoc1)CO)OC 29530,CN=c1nc(C(=O)NC2CC2NC(=O)CCn2cnnn2)cc(C)[nH]1 29531,C1(CNC(C(C)P(C)(C)=O)=O)CC2CCC(C1)N2C(C1CCCCCC1)=O 29532,C=CCCC(C(=O)N(C)Cc1cn(C)cn1)NC(=O)CC1CCCCN1C 29533,c1(-n2cc(CN(C(COc3ccn(C)n3)=O)C3CC3)nn2)cccnc1Br 29534,C1(COC)CC(Cn2cc(C3CC3)nn2)N(C(=O)C(C)(C)F)C1 29535,C(N=c1[nH]c(=NCC2CC3(CCC3)C2)c2[nH]ccc2[nH]1)c1nn(C)c(C2CC2)c1 29536,c1(C(N2CCC(C3(C(F)(F)F)N=N3)C2)=O)cc2ccsc2s1 29537,c1(CC)ccc(C(=O)NC2CCC2NC(=O)CCc2nnc(O)nc2O)cc1N 29538,N1(C(=O)Cc2ccc(Br)cn2)CC2CCC(C1)C2NCc1c(F)cccc1Cl 29539,N1(C(CC(C)C2CCCCC2)=O)CCC2(CC1)CN(C(=O)C=CI)CCO2 29540,c1(C(C(C)N)N(C(=O)CCn2cc(CC(C)(C)C)nn2)C)cccnc1.CO 29541,c1(C(N2CCC(NC(CS(CC)=O)=O)C2C)=O)ccc(Br)cc1OC 29542,N1(C(C2(CC)CC(F)(F)C2)=O)CCOc2cccc(C(=O)O)c2C1 29543,C1(O)(C(C(=O)Nc2ccc(OCc3ccco3)cc2)OC)CCCCC1 29544,N1(C(C2OCCN(C)C2)=O)CC(NC(c2cccnc2Cl)=O)CC2(CC2)C1 29545,C1(CNC(C2CCN(c3ccccc3Cl)C2)=O)COCCN1C(c1cnns1)=O 29546,C(C(COC)C(=O)NC(Cc1ccco1)C(=O)NCCC1CC1C)OC 29547,C(C)(CO)(C(=O)N1CC(C)(C)C1C(C)C)NC(c1c(OC)nsc1)=O 29548,N1(C(c2c(C)sc(O)n2)=O)CC(C)C(NC(c2cc[n+]([O-])cc2)=O)C(C)C1 29549,c1(C(=O)OCC)cc(C)c(F)c(S(=O)(=O)Nc2c(C)ccnc2OC)c1 29550,C1(NC(=O)C(C2CCCO2)C2CC2)CCCCC1CNC(=O)C(F)(F)C1(O)CCC1 29551,c1(CC(=O)NCCOCCNC(COC(CC)C)=O)csc(Cl)n1 29552,c1(CNS(C)(=O)=O)cccc(C(=O)NCC2CC(NC(C3(C)CCC3)=O)C2)c1 29553,C(=O)(CCCCCC)N(C1CC(NC(CSCC#C)=O)C1)C 29554,Cc1ncc(F)c(=NCC2(C)CCN(C(=O)CC3CCC(C)C(C)C3)C2)[nH]1 29555,N(C(=NCCOC1CC1)NCC1(CO)COCCN1C)Cc1cc(C)oc1 29556,C1(NC(C)=O)CCC(C(=O)N(C2CC(C#N)C2)CCO)CC1 29557,c1(CC(N2CCC(CNC(CC(C)C)=O)CC2)=O)ccc(C#N)nc1 29558,C=CCN=C(NCc1nnn(C)c1C(F)(F)F)NCC(CO)C(C)C 29559,Cc1ccccc1CC(C)C(=O)NCC(C(C)C)NC(=O)CN(C(=O)C(C)C)C 29560,C1(CNC(C2(N(C)C)CCCC2)=O)C2CC1N(C(C1CCS(=O)CC1)=O)C2 29561,C(c1ccc(C)c(Cl)c1)=CC(=O)NCC1C=CC(NC(Cc2ccc(C)s2)=O)C1 29562,c1(CCNC(=O)OC(C)(C)C)c(C)nc(O)nc1O.C1(c2ccoc2)C(=O)N1 29563,C1(C(=O)OC)COCCC1NC(C1CSCC1C)=O 29564,N1(C(c2c(OC)n(C)nc2)=O)CC2CC(NC(C3CCS(=O)(=O)CC3)=O)C(C2)C1 29565,c1(CC(=O)NC(C2CCN(C(c3ns[nH]c3=O)=O)C2)(C)C)c[nH]c2cnccc12 29566,S(=O)(=O)(c1ccc(NC2CC(C3CC3)C2)c(Br)c1)NC1(CC(C)C)CC1 29567,N1(S(C)(=O)=O)CCC(NC(c2ccc(C(=O)C3CC3)cc2)=O)C1c1ccccc1 29568,C1(C(C)CNC(=O)C=CCO)CCN(C(C2CCC23CCC3)=O)CC1 29569,n1(C2(Oc3ccncc3)CC2)ccc(=Nc2ncnc3ccsc23)[nH]1 29570,Cc1cnc(N2CCSCC2C)c(S(=O)(=O)N2CCOC(C3CCCC3)C2)c1 29571,C1(C)(CNC(CC(C)(O)c2ccccc2)=O)CCCN(C(C2(CF)CCC2)=O)C1 29572,C(=O)(C1=CCC(NC(c2ccc(C#N)n2C)=O)C1)NC1C(C=C)COC1 29573,C1(C(=O)NC2C(C)C2C)(CO)CCN(C(C2CN(C(N)=O)C2)=O)C1 29574,C1(CC(=O)O)COC(C)(C)CO1.C(=O)(C(C)CC)N(CC(CC)NC(=O)CC1(O)CC1)C(C)C 29575,C(=O)(CCS(N)(=O)=O)N1CCCC(CCC(=O)N(C)Cc2onc(CC)n2)C1 29576,N1(C(C(CC=C)CC)=O)CCC2(CCCN2C(=O)CCCOC(C)C)C1 29577,CCCCC(CNC(c1ccc(OC(C)CC)cc1)=O)NC(C1CCCCO1)=O 29578,c1(CC(=O)NC2CCN(C(=O)C3=COCCO3)CC2O)ccc2c(c1)NC(=O)C2 29579,CC1(C)CN(C(=O)CC2CC(=O)NC2=O)CC1NC(=O)Cc1ccc(O)cn1 29580,C1(CNC(C(C(C)C)N(C)C)=O)CN(C(=O)C=CC(F)(F)F)CCC12CCC2 29581,C1(C(N2CCC(NC(c3c(OC)oc(C)n3)=O)C2)=O)CC(c2cnn(C)c2)=NO1 29582,C1(NC(CC2(COC)CCCC2)=O)CC(C)N(C(c2ncncc2Cl)=O)C1 29583,C12CC(O)CN1C2=O.c1(C2(CNC(=O)CO)CC2)ccc(C(F)(F)F)cc1 29584,C(=O)(C1=CS(=O)CCC1)N1CCC(NC(C(C)NC(=O)CC(C)(C)C)=O)C1C 29585,N1(CC(=O)N(C)CC2(CNC(C3CC=CC3)=O)CC2)CCSC2CCCCC12 29586,C=C1CC2(C1)CC(C(N1CC(OCCNC(C3CCOC(C(C)C)C3)=O)C1)=O)C2 29587,C(=O)(CCCNC(c1cc(Cl)c[nH]1)=O)N(C1(C(=O)OC)CCC1)C1CC1 29588,N1(C(C(C)(C)Nc2ccccc2)=O)CCN(C(C2CC(F)(F)C2)=O)CC(O)C1 29589,N1(C(CN2C(C)CC2)=O)CCC2(CCC2)C(NC(=O)Cc2csc(S)n2)C1 29590,N1(C(c2c(COC)nc(=N)[nH]c2)=O)CC2CC1CN(C(=O)CS(N)(=O)=O)C2 29591,CC(CC(=O)N1CCCC1CN(C(=O)C(C)(C)c1ccns1)C)P(C)(C)=O 29592,N1(C(C2C(=C)CC2)=O)CCC2(CCC2)C(CNC(c2ccc(N)cn2)=O)C1 29593,O=S(=O)(c1ccc2c(c1)OCCCO2)NCC1(CF)CC2(CCC2)C1 29594,CCC(C)C(C(=O)NCCOCC(=O)NCCc1cnc(C)o1)OC 29595,N1(c2ccnc(C(CC)C)n2)CCCCC(CNC(c2cccn2C)=O)C1 29596,c1(C(=O)NC2CC(C(N(CC(F)(F)CO)C)=O)C2(C)C)cnn(C)c1C#N 29597,N1(C(C2(CC)CC2(F)F)=O)CCCC(N(C(=O)CC2(OC)CCOCC2)C)CC1 29598,Cc1noc(CCC(=O)NC(C2CCN(Cc3nc(C(F)F)no3)C2)C)n1 29599,N1(S(c2c(C)nc(C)s2)(=O)=O)CCCC2(CCS(=N)(=O)C2)C1 29600,C1(C(=O)NC2CC(O)(CNC(C3(CC(C)C)CC3)=O)C2)CCS(=O)(=O)N1 29601,CC1(NC(C2CCC(NC(C3CCCC3F)=O)CC2)=O)CC(F)(F)C1 29602,c1(CCC(=O)N(C2CCN(C(c3cc(C(C)=O)oc3)=O)C2)C)cnn(C)c1C 29603,c1(C(=O)NCC(C)NC(c2c(CC)nco2)=O)ccc(OCC(C)C)cc1 29604,c1(C(N2CCOCC(NC(CC=CC)=O)C2)=O)cnn2c1C(C)CCC2 29605,c1(C(=O)NCC2(F)CCC(CNC(C(CC#C)O)=O)C2)cccc(C2CC2)c1Cl 29606,c1(OC)ccc(C(C)=CC(N2CC(OC)CC(NC(C3(O)CCC3)=O)C2)=O)cc1 29607,c1(C(=O)OC)c(C)[nH][nH]c1=NC(=O)c1csc(NCc2cc(OC)cc(F)c2)n1 29608,Cc1ccncc1C=CC(=O)NCC(CC(C)C)NC(c1ccnc(C)c1C)=O 29609,C12(NC(C=Cc3ncc(C)[nH]3)=O)CCOCC1CN(C(c1nccnc1C)=O)C2 29610,c1(N2CC(CCOC)OCC2)nc(NC(c2cccc(F)c2)C)c2ncsc2n1 29611,S(=O)(=O)(CCCCCl)NC1CC(C(=O)Nc2cnccc2C(F)(F)F)C1 29612,N1(C(CC(CC)(F)F)=O)CCCC12CCN(C(c1cnc3ncc(Cl)cn13)=O)C2 29613,C1(C)(CNC(Cc2n(C)nnc2)=O)COCCN(C(C2CCC3CCC2O3)=O)C1 29614,N1(C(CC(COC)NC(c2cc(CC)no2)=O)=O)CCC(O)C(C)(C)C1 29615,Cc1cccc(C)c1OCC(=O)NCC1CC(NC(C2(C)CC3CCC2C3)=O)C1 29616,C12(NC(C3C4CN(C(C5OCC(C)(C)C5)=O)C3C4)=O)CCC(CC1)OC2 29617,CC1(OCC(=O)NC2(C)CC(F)C2)CN(C(=O)COCCC(O)CO)C1 29618,C1(NC(=O)CC2CC=CC2)CN(C(C2CC2F)=O)CC12CCC2 29619,C1(CNC(C2(C(N(C)C)=O)CC2)=O)CC2CCC1N2C(=O)Cn1cc(CO)nn1 29620,CC1CCCCC1(C)C(N1CCC(CF)(NC(c2ccc(C(N)=O)[nH]2)=O)C1)=O 29621,N1(C(c2n(CC)ccn2)=O)CC2CCC1CN(C(=O)C(c1ccc(O)cc1)=O)C2 29622,c1(C(N2CC(NC(c3c[nH]c(=N)s3)=O)C(CO)CC2)=O)cccn2nnnc12 29623,C(CCS(N)(=O)=O)NC(C=C(C)CNC(C1CC1(Cl)Cl)=O)=O 29624,C12(OC(C)(C)C)CC(C1)C(=O)N2.C1(C(=O)OC)(C(=O)OC)CC1C 29625,N1(C(=O)Cc2cncnc2O)CCC(NC(C23CCN(CC2)C3)=O)C(CO)CC1 29626,Cc1c[nH]c(CC(N)=O)c1C(=O)NCC1CCC(O)CC1 29627,N1(C(C2(CC)CC2)=O)CCC2(CC1)CCN(c1ncnc3c(C)cccc13)CC2 29628,c1(C(N2C(C)CC(CNC(CCc3cc(C)no3)=O)C2)=O)ccc(N)c(O)c1 29629,C1(NC(CCCCOC)=O)CC2CCC(C1F)N2C(C1CN(CC(F)(F)F)C1)=O 29630,c1(OC)cccc(CC(=O)NC2CC(CO)N(C(c3cnc(C4CC4)s3)=O)C2)n1 29631,C#CC1CN(C(c2ccc(OC)c(F)c2)C(=O)NCC=C)CCO1 29632,C1(C(=O)NCC(C)CC2CCCC2)CCCN(C(c2ccc(C(F)F)o2)=O)C1 29633,N1(C(CCC(N)=O)=O)CC2CC1CC2NC(=O)C#CC1CCC1 29634,C1(c2scc(C)n2)CCCN(C(=O)CNC(=O)CCCn2cccn2)C1 29635,C(c1ccoc1)=CC(=O)NC(C(=O)NC(C(=O)OCC)C1CC1)C1CCC1 29636,C#CCCC(=O)NC1CC(OCC(=O)N(C(C)C(C)CC)C2CC2)C1 29637,Cc1ccc(C(O)C(=O)NC2CC(NC(c3cnc(O)n3C)=O)C2)cc1 29638,Cc1nn(CC(N2CC3CCC3(NC(=O)CCCNC(N)=O)C2)=O)c(C)c1Br 29639,CC(C)CC(CNC=O)CC(=O)NC1CCC1NC(c1ccc(CO)cc1)=O 29640,CCCC(C(=O)N=c1ccn(C(C)C)[nH]1)NC(=O)CCCSC 29641,C1(C(=O)NC2CC(CCNC(c3c(C#C)cnn3C)=O)C2)CC2(COCCO2)C1 29642,CCS(=O)(=O)CC(=O)NC1CCC(C)(CNC(=O)CS(=O)(=O)N(C)C)C1 29643,C(=O)(C1=CCC(C(F)(F)F)OC1)NC1C(NC(C=CCN(C)CC)=O)CCC1 29644,CC1CC(CCNC(c2ccc(C(N)=O)[nH]2)=O)CCN1C(c1ccoc1)=O 29645,N1(C(c2c(OC)noc2C)=O)CCCN(C(=O)CN2CC(=O)NC2=O)CCC1 29646,C1(NC(CC=C)=O)(CC)CCN(C(c2cccc(C(C)(F)F)n2)=O)CC1 29647,c1(C(=O)NCC=CCNC(C2C(CC)CCC2)=O)ccc2c(c1F)CCC2 29648,C1(NC(=O)NC2C(c3n(CCOC)ccn3)OCC2)CC2CCC1O2 29649,c1(C(=O)NC(c2ccn(C)n2)C)ccc(C(=O)O)cc1F 29650,C1(C(=O)NC2(CN(C)C(c3nccn3C)=O)CC2)C2CCC1(c1ccccc1)C2 29651,Cc1ccc2c(c1)C(NCCCC(N)=O)C(C)C2 29652,C1(NC(CCCCCCCCC)=O)CCN(C(=O)C(C2CC2)SCC)CC1(C)C 29653,N1(C(C2C(CCC)CN(C(=O)C(C)CC(N)=O)C2)=O)CC2(C1)CC(C)(C)C2 29654,N1(C(C(CC)SC)=O)CCc2sc(CNC(C3(OC)CS(=O)(=O)C3)=O)nc2C1 29655,N1(C(c2c(C)n(C)nc2)=O)CC2C3CCC(C2C1)N(C(=O)CS(=O)(=O)C(C)C)C3 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29674,C12(C(=O)NCC3N(C(C=CC(CC)=CC)=O)CC3)CCOC1CCOC2 29675,c1(CC)cc(C(=O)NCC2CCCN(C(=O)C(=O)N(C)C)C2)oc1CC 29676,c1(C(=O)NC(C(C)NC(C2CCCN(CC(F)F)C2)=O)C)cnc2[nH]ncc2c1 29677,c1(CC(=O)NCC2(NC(=O)CCC3CCCCO3)CCOC2)cccc(Cl)c1 29678,C1(CNC(=O)CCC2CC2(Cl)Cl)CC2(CCC2)CN1c1nc2ccccc2o1 29679,Cc1cncc(-c2cn(CC3CCN(C(c4oc(C5CC5)nc4C)=O)C3)nn2)n1 29680,CC1CCc2nnc(C(N3CCN(C(C)C(=O)N(C)C)CC3)=O)n2C1 29681,C1(NC(c2n(C)ncc2)=O)CC2CCC1(NC(c1cc(C(N)=O)co1)=O)C2 29682,N1(C(C2CC(C(C)=O)C2(C)C)=O)CC2CCC(CNC(=O)Cc3cnsc3)(C2)C1 29683,C1(NC(c2cn(CC)nc2C)=O)CC12CCN(C(=O)Cc1nc(=N)[nH][nH]1)C2 29684,S(=O)(=O)(c1cc(Cl)ccc1Cl)NC1CCCN(C(CSC2C(=O)OCC2)=O)C1 29685,c1(OC)ccc(CC(C)C(=O)NC(C)CCNC(=O)Cc2sccc2C)cc1F 29686,C1(NC(C2CN(CC)C(=O)C2)=O)CC2CCC(C1C)N2C(c1cc(C)c(C)o1)=O 29687,C1(C(N(C2CCC(NC(C3CCC(CC)O3)=O)C2)C)=O)C2CCC3C(C2)CC13 29688,C(C)(C)(CC(F)C(=O)NC)NC(C(COC)COC)=O.C(C(C)C)NC 29689,C(CC1=CCN(C(C2(C)CCCO2)=O)CC1)NC(C(C(C)C)n1cc(C)nc1)=O 29690,c1(C(=O)NCC2CC(O)CN2C(=O)CCOC2CC2)cncc(Cl)c1Cl 29691,N1(C(c2ccc(S(C)(=N)=O)cc2)=O)CC2C3CCC(C2C1)N(Cc1cccs1)C3 29692,c1(OCCC)cccc(CC(=O)NC(C)C(C(C)C)NC(c2cncnc2)=O)c1 29693,N1(C(=O)NC2C(CC)CCCN2)CCCC(c2ccccc2)C1C 29694,C(=O)(C1CCCn2nccc21)N1CCC(CCc2cn(C(C)CO)nn2)CC1 29695,Cc1cc2c(cc1C)C(N(C(c1cc(F)cc(C)c1C)=O)C1CC1)CCCO2 29696,N1(C(c2cc(OCC)n[nH]2)=O)CCC(C(=O)Nc2cccc(Cl)c2)C12CC2 29697,n1(CC(=O)NC2CC(C(=O)NC(C3(CO)CC3)C)C2)cnc(C#N)n1 29698,c1(C(N2CC(CCNC(c3cc(C)c(N)cn3)=O)C2)=O)ccc2c(n1)OCCO2 29699,C(CC(Cc1ccccc1)NC(C1(Br)CC1)=O)NC(c1cnns1)=O 29700,c1(C(N2CC(CCNC(C3CC=C(C)CC3)=O)C(C)C2)=O)cccc2nc[nH]c12 29701,C1(NC(C(C)(C(C)C)OC)=O)CN(C(=O)CN(c2ncccn2)C)CC2(CC2)C1 29702,C1(C(=O)NC(C(C)F)C)CC2CC1CN(C(=O)CC1CCC(C)(C)O1)C2 29703,C(=O)(C(CCC(C)C)NC(c1cnn(C)c1Cl)=O)N(CCCSC)C 29704,c1(C(N(CCC(C)NC(CC)=O)C)=O)cccc2c(I)n[nH]c12 29705,C(c1ccc2c(c1)OCCO2)=CC(N1CCCC(N(C(C(CC)CC)=O)C)C1)=O 29706,C#CCCCCCC(=O)N1CC2(CC(C(=O)NC3CC(=O)N(C)C3=O)CO2)C1 29707,c1(C(=O)NC2C(NC(C(C)OCC(C)C)=O)CCC2)cc(C2CC2)ccn1 29708,Cc1nnc2cnc(C(=O)NC3CC(CNC(c4ccc(Cl)c(Cl)c4)=O)C3)cn12 29709,c1(OCCN(C)C)ccc(S(=O)(=O)N2CCCC(c3noc(C4CCCO4)n3)C2)cc1 29710,C1(C(=O)NC2C(C(=O)NC(c3c(C)nns3)C)CC2)CCC(C)CC1 29711,c1(C(C)C)conc1C(=O)NC(C)CC(=O)NC1COCC1CN(C)C 29712,C(=O)(C(CC1CCC1)NC(c1cc(F)c[nH]1)=O)N(C)CCOCC1CC1 29713,n1(CC(=O)NC2(C)CC(NC(C(CCOC)C)=O)C2)cc(C)c(O)nc1=O 29714,C1(NC(=O)NCc2cc(NC(C)=O)c(OC)cc2)CN(C(C)=O)C2CCCC12 29715,C(=O)(CCCCC(F)(F)F)N1C(C)CC(CCNC(=O)COCP(C)(C)=O)CC1 29716,c1(CNC(C(C)C#N)=O)cccc(CNC(=O)CC(C2CC2)C2CC2)c1 29717,C1(C2CC2)(NC(C2CCC(NC(Cc3c(C)ccs3)=O)C2)=O)CCCC1 29718,CC1(C)CN(C(c2ccc(OC(F)(F)Cl)cc2)=O)CC1c1ccc(Br)cc1 29719,Clc1ccccc1Cn1nnnc1N1CCN(CCSc2ccccc2)CC1 29720,C(=O)(CCN=[N+]=[N-])NC1(CCC(=O)NCC(COC)O)CCCC1 29721,C1(NC(c2nc(C)oc2C)=O)CCN(C(=O)C(F)C(C)C)CC1CO 29722,C1(CNC(c2cc(O)ccc2I)=O)CCN(Cc2c(F)cncc2F)CC1(F)F 29723,c1(C(N(CC(C)C)CC(=O)NCC2CC(=C3CCC3)C2)=O)ncccc1N 29724,N1(C(C(C)(C2CCC2)NC(CC(C=C)(C)O)=O)=O)CC2CC=CCC2C1 29725,CC(CC(=O)NCC1CC12CC2(F)F)C(C)(C)NC(=O)C=C1CCOCC1 29726,C(=O)(C(C)(C)C(F)(F)F)N1CCC(OCCNC(c2c(C)n(C(C)C)nc2)=O)C1 29727,CCC(CNC(=O)CC(C)C1CCCO1)(CC)NC(=O)C(C)CC1CCC1 29728,Cc1nn(C)c(C(=O)NCC2CN(C(=O)COC(F)F)CCCO2)c1Cl 29729,S1(=O)(=O)c2ccc(Br)cc2NCCCN1CC=C.S(=O)(=O)(C1CC1)NCCO 29730,C=CC1OCCC1C(N1CCN(CC2(NC(=O)Cn3ccnc3C)CC2)CC1)=O 29731,C1(NC(c2cn(C)c(=O)cn2)=O)COC2CN(C(=O)CC(C)(C)O)CC12 29732,C1(CNCC2N(C(c3cc(C)cc(O)c3)=O)CCC2)COc2ccccc2O1 29733,c1(C(=O)NCC2N(C(C3=C(C)OCC3)=O)CCOC2)ccc([N+](=O)[O-])c(F)c1 29734,C12CCN(C(C)C1)C(=O)C(=O)N2.n1(CC)nc(C(N(C)CC2CC2)=O)cc1C1CC1 29735,C=CCC(C(=O)NC1CCCN(C(c2snnc2CC)=O)C1)OC 29736,C(=O)(C(C)(C)C(F)F)N(C)CC1CN(C(C(C)SC)=O)C1 29737,CCC(C)(CNC(=O)C(C1CCCCC1)C)NC(c1occc1C1CC1)=O 29738,c1(CNC(C2CC(NC(COCCOC)=O)C2(C)C)=O)ccc(O)c(C)c1 29739,c1(C(C)=O)ccc(C(N2CCCC(C)C2)=O)cc1F.C1(=O)C(=O)NCCN1CC 29740,c1(NC(CC(C=CC)OC)=O)ccc(S(=O)(=O)CCNC(=O)OC(C)(C)C)cc1 29741,C1(COC)CN(C(c2cc(F)c[nH]2)=O)CCN1C(=O)CCCc1ccc(O)cc1 29742,N1(C(C2CC(SC)C2)=O)CC2CC(NC(=O)CC3(O)CCCC3)CC(C2)C1 29743,c1(C2CCN(CC3CCN(Cc4c(Cl)c[nH]n4)CC3)C2)cccc2c1OCO2 29744,c1(OC)ccc(OC(F)(F)F)cc1C(=O)NCC1CC1NC(=O)CCCCCF 29745,c12sc(C)cc1NC2=O.N1(CCNC(CN(C(=O)OCC)C)=O)CCC(C)C1 29746,Cc1cc2ccc(C(N3CCC(NC(c4[nH]c(O)nc4C)=O)CC3C)=O)cn2c1 29747,N1(C(C2N=C(C)SC2)=O)CCOCC(CNC(=O)Cc2cccc(N)c2)C1 29748,C1(C(N2CC=CC(C(=O)NCCC3CC(F)(F)C3)C2)=O)C2CCC(F)(F)C12 29749,C(=O)(C(C)CC(F)(F)F)N(CCNC(c1n(CC)nnc1C)=O)C1CC1 29750,c1(C(=O)NC(C(C)NC(c2c(C)cc(F)cn2)=O)CO)cnc2c(c1)COCC2 29751,C1(C(=O)NCCOCCCNC(=O)Cn2cccc2)CC(=O)N(c2cn[nH]c2)C1 29752,c1(C(C)O)ncc(C(N2CCCC2C(C)(C)NC(c2nsnc2O)=O)=O)s1 29753,c1(NC(=O)Nc2cc(C)c(Br)cn2)cc(C(F)(F)F)cc(S(C)(=O)=O)c1 29754,C1(C)(C(=O)NCC(C)(CO)NC(CC2CC(=C)C2)=O)CC(=O)N(C)C1 29755,c1(C(N(CCCNC(C(CC)C)=O)Cc2ccccc2)=O)nc(C)ccc1F 29756,c1(C(=O)NCCc2cn(CC(C)(C)O)nn2)snc(-c2ccccc2)c1Cl 29757,CCCCC(O)C(C)C(=O)NCCCC(=O)N(CC(C)OC)C 29758,N1(C(CCc2cnc(C)s2)=O)CC2C(CNC(c3cc(F)cs3)=O)C2C1 29759,C1(C)(CC)NC(=O)N(CC(=O)NC(C)C(C)NC(c2c(Cl)n[nH]c2CC)=O)C1=O 29760,C(=O)(C(C(C)(C)C)NC(C1CCC2(CCC2)O1)=O)N1CCC(C)CC1 29761,CC(C)C(F)(F)CC(=O)NCC1(C)CN(C(C2CCOC2C)=O)CCO1 29762,C#CCCC(O)C(=O)N(CCN(C(C1(C)CCCNC1=O)=O)CC)CC 29763,Cc1cc(C)n2nc(C(N3CCC3CNC(=O)C3=CCCCO3)=O)cc2n1 29764,C1(CNC(c2scc(C)c2C)=O)CN(C(c2ccc(C(F)F)o2)=O)CCC1C 29765,N1(C(=O)NC(c2cnn(C)c2)C(C)C)CCOC(C)(C(F)F)C1 29766,c1(-n2c(CC(C=C)C)nc(C3CCCCC3)n2)ccnc2ccccc12 29767,C1(NC(CCC(=O)OC(C)(C)C)=O)CC2CC1CN2C(c1cnc(C(N)=O)s1)=O 29768,CC(O)C(C(=O)NCC1(CO)CC1)NC(C1CC(F)(F)C1)=O 29769,c1(-c2nc(CC)nn2-c2cccc(NC(C)=O)c2)cnn2ccc(O)nc12 29770,N1(C(C2CCn3nccc3C2)=O)CCCC2(CCN(C(C34CC(F)(C3)C4)=O)C2)C1 29771,C=CC1(CC(N2CCC(NC(c3cscc3C)=O)C(CC)C2)=O)CCOCC1 29772,C1(NC(C2CN(C(=O)OC(C)(C)C)CCO2)C)CCCN(C(C)(C)C)C1=O 29773,CCCCCCC(=O)NC(CNC(=O)CCc1ccc(Cl)c(Cl)c1)C(C)C(C)C 29774,c1(NCC23N(C(=O)OC)CC(C2)OC3)nc2ccccc2nc1C 29775,c1(C(=O)NCCCC2N(C(C(CCCC)O)=O)CCC2)c(C)nc2sc(C)cn12 29776,C(CCC(C)C(=O)NCC12CC(CO1)N(C(=O)CCc1nc(O)n[nH]1)C2)OC 29777,c1(C(=O)NC(C2CCCCO2)C)cc(CNC(C2COCOC2)=O)nn1C 29778,C1(CNC(CC(C)n2ccnc2)=O)C(C)CCCN1C(=O)CC1(O)CCCOC1 29779,c1(NC(C2CSCCN2C(c2ccc(Br)s2)=O)=O)cccc(O)c1F 29780,c1(CN2C(C(=O)Nc3ccc(CC)nc3)CC(O)C2)ccc(C#N)nc1 29781,N1(C(C2(CC)CC2)=O)CCCC2CN(C(=O)C(=O)Nc3ccc(C)cc3)CC12 29782,C(C(CC1CC1)C(=O)NCCCCOC(=N)O)NC(C(C1CCCC1)OC)=O 29783,n1(CC(C)CO)nc(-c2ccc(Cl)nc2)nc1C1CCC(=O)N1C(C)(C)C 29784,N1(C(c2ccc(C)nc2O)=O)CC2OCC(NC(=O)CCC3(C)CC3)C2C1 29785,c1(C(=O)NCC(C)NC(Cn2c(C)nc(C)n2)=O)ccc2c(O)nc(C)nc2c1 29786,CCC(C#N)(CC)C(=O)NCC(O)CNC(C1(OC)CC1)=O 29787,C(=O)(CCCCCCNC(C1CCOC1(C)C)=O)NCC(C(C)O)C 29788,c1(C(=O)NCC(CC)NC(C2(O)CCCCC2)=O)cn(C)nc1C(C)(F)F 29789,N1(C(C2CC(NC(CCC3(C#N)CCC3)=O)C23CCC3)=O)CCOC2COCC12 29790,C1(COC)(CNC(c2csc(C)c2N)=O)CCN(C(=O)C(C)c2ccsc2)CC1 29791,N1(C(C(C2(C)CC2)NC(C(COC)C)=O)=O)CC2(CC(C)CO2)C1 29792,C1(OC)CC2CCC1CC2C(N1CCC(N(C)C(c2ccc(C)c(C)c2)=O)C1)=O 29793,c1(C(N(C2C(NC(C3(C=C)CC3)=O)CCCC2)C)=O)cc(C)nc(O)c1 29794,N1(C(C2COCCO2)=O)CC2C(NC(C3(C(F)(F)F)CC(F)(F)C3)=O)C2C1 29795,C(N=c1cc(CC2CC2)nc[nH]1)C1(F)CC(NC(CC(C(C)C)O)=O)C1 29796,c1(CNC(C(=O)N(C)CCc2ccc(C#N)cc2)=O)sccc1S(C)(=O)=O 29797,c1(OC)ccnc(C(=O)NCC2CCCCN(C(c3csnc3C)=O)C2)c1F 29798,c1(C(=O)NCC(C)CN(C)C(c2cc3nc[nH]c3cn2)=O)cncc2sccc12 29799,N1(C(C)C)CCCC(C(=O)NC2CC3(CC3)C2)C1.N12CCN(CC1)CC2 29800,C1(C(N2C(C=C)CC2)=O)(NC(=O)CCOC(C)=O)CCCC1C 29801,CN1CCN(C(C2CCC2(F)F)=O)C(C(=O)NCC2(CO)CCC2)C1 29802,c1(N2CC(=C(CNC(C3C=CCCC3)=O)F)C2)ncc2cccnc2n1 29803,N(C(=NCCN1CCCC1)N1CCCC2(CC2)C1)Cc1oc(CC)c(C2CC2)n1 29804,C1(NC(c2nccc(C)n2)=O)CC(CNC(=O)Cc2nonc2C)C12CCC2 29805,C(=O)(CC(C(=C)C)OCC)NCC1C(C(=O)NC2(CC=C)CC=CC2)COC1 29806,c1(NC(=O)Nc2cnsc2)ccc(C(=O)Nc2cccc(-c3nn[nH]n3)c2)cn1 29807,C1(C)(C(=O)NCCNC(C(c2ccc(Br)cc2F)C)=O)C(C)(C)C1(C)C 29808,C1(NC(C=C(C)C(C)C)=O)C2CC1N(C(=O)CC(c1ccccc1)NC(N)=O)C2 29809,C(N=c1[nH]c(N(C)CC2CCCO2)nc(=N)[nH]1)c1c(C)ccnc1 29810,CCCC(C#N)C(=O)NCC1(F)CC(NC(=O)Cc2cncn2C)C1 29811,C(=O)(CC(C(F)(F)F)NC(=O)CNC(=O)C(C)(C)C)NCC(=C)Br 29812,N1(C(c2cc(COC)no2)=O)C(C(=O)NCc2snnc2C)CCC12CC2 29813,c1(OC)ncnc(N2CCC3(CC3C(=O)Nc3ccc(O)cc3C(N)=O)C2)c1C 29814,N1(C(CC2N(C)CCC2)=O)CCC(C2CCCN(C(c3ccc(Cl)o3)=O)C2)CC1 29815,N1(C(c2cc(CCC)ncc2)=O)CC2CCC(C1)N2C(=O)Cc1cnn(C)c1 29816,C1(C(N2CCC(NC(c3cnn(C)c3Cl)=O)C2)=O)Cc2ccccc2CO1 29817,Cc1nn(C)cc1C(=O)N(C)CCNC(=O)CN1CCCCC1=O 29818,CCC(C)C(CN(C)C)NC(c1ccc(CNC(=O)C(C2CCC2)OC)s1)=O 29819,CC(C)CCCC(C)C(=O)NC1C2CC3C(C2)C13C(=O)N(C(CO)C1CC1)C 29820,c1(C(N(C2CCN(C(C(=CC3CCCC3)C)=O)C2)C)=O)nc(Cl)c(Cl)s1 29821,C1(C(=O)Nc2cccc(C3CCCCC3)c2)CC(F)CN(C(c2ncc[nH]2)=O)C1 29822,CCCCC(=O)C(=O)NCC=CC(N1CC(S(C)=O)C1)=O 29823,C1(CCOC)(NC(=O)C(O)CCSC)CCN(C(=O)CN(C2CCC2)C)CC1 29824,N1(C(CC(CC)SC)=O)CC(NC(c2cc(C)n(C)c2C)=O)CC1(C)COC 29825,C(=O)(CS(=O)(=O)C(C)(C)C)N1C2(CNC(CC(CC)C)=O)CC(C1)C2 29826,CCCC(CC)C(=O)N1CCC(CNC(c2csc(CC)n2)=O)C12CC2 29827,C(=O)(CCC(F)(F)C(=O)N1CCCCC1CNC(C1(C)CNC(=O)C1)=O)OCC 29828,N1(CCNC(C=CC2(C)COC2)=O)CCN(C(=O)CC2CCNC2=O)CC1 29829,Cc1nc(C(C)(C)C)sc1C(=O)NCC1(NC(C2CCCC2)=O)CCCC1 29830,C(=O)(CC(O)CC(C)(C)C)N1CCC(N(C(c2cncc(C)c2)=O)CC2CC2)C1 29831,c1(C(N2CC(F)CC(NC(=O)C3=COCCO3)C2)=O)cccc2c3c([nH]c12)CCC3 29832,C(CO)(CCF)NC(C(C)N(C(=O)C=C1CCC1)C1CC1)=O 29833,Cc1cccc2c1c(CNC(c1cc(F)c(Br)c(F)c1N)=O)cn2C 29834,c1(CCNC(C(C2CCCC2)NC(C2C(C)(CC)C2)=O)=O)ccccc1 29835,Cc1oc(C#N)cc1C(=O)NCC1(C)CCN(C(C2CCCC(C)CC2)=O)CC1 29836,CCC(CC(=O)N1CCCC1(C)CNC(=O)CC1(C)CCOCC1)C(C)(C)C 29837,CC1(C)OCCC1CC(=O)NC1CCCC1NC(c1ncccc1O)=O 29838,N1(C(c2c(C)n(C)cc2)=O)CCCCC(NC(c2ccc(CO)s2)=O)C1 29839,Cc1ccc(O)nc1CNC(C1CN(C(=O)CC2C(C)(C)C2(C)C)CC1F)=O 29840,N1(c2cc(=NC)[nH]cc2[N+](=O)[O-])CCC2(CC1)COC(CNC(=O)C(C)OC)C2 29841,N1(C(CC(=O)OCC)=O)CCC(NC(=O)Cn2nnc(C)n2)CC(C)(C)C1 29842,N1(C(CC=CC)=O)CC2CCC1C1CN(C(=O)CCCOCC)CC21 29843,C1(C(=O)NC2CN(C(c3c(C)onc3)=O)CC2(C)C)Cc2ccccc2S1 29844,C(C1=NOC2CCCC12)NC(C(=O)NC(COc1ccc(C)cc1)C)=O 29845,C=C(C)C1CN(C(=O)CN(C)C(C2CCN2C(C)(C)C)=O)CCO1 29846,c1(C(N(C2CC(NC(c3cnn(C)n3)=O)C2)C)=O)cc(C(F)(F)F)n(C)n1 29847,CCCC(CC)C(=O)NCC1CCC1NC(=O)COCC1CCCC1 29848,C12(C(=O)NCC(CC)(C)OC)CC(CN1C(=O)CCOCC(C)(C)C)C2 29849,C(=O)(CC(C)P(C)(C)=O)NCCCN(C(CSCC(=O)OC)=O)C(C)C 29850,C(=O)(C1=CCCN(C(C2CCC=CCC2)=O)C1)NCc1n(C)nnn1 29851,CCC(C)(CCNC(=O)C=Cc1c[nH]cn1)NC(=O)CCCc1ncco1 29852,N1(C(C(c2ccc(C)cc2)C)=O)CC2=C(C1)CN(C(c1c[nH]cc1C)=O)C2 29853,C12(C(=O)NC3(C(=O)OCC)CC3)CCC(CN(C(=O)C3=NOCC3)C1)C2 29854,CCCC(C)(CCC)C(=O)NC1CN(C(=O)CCN(C)C(C)=O)CC1C1CC1 29855,C(N=c1nc(O)c(Br)c[nH]1)C1CCCC(NC(c2ccc3nncn3c2)=O)C1 29856,c1(C(N2C(CNC(C3CC(=O)N3)=O)CC(C)(C)C2)=O)cnc(O)c2ncccc12 29857,Cc1nc2ccnn2c(C)c1C(N1CCN(C(c2cnc(O)n2C)=O)C(C)C1)=O 29858,Cn1cnc(C(O)CNC(=O)CC2(NC(C3CC(F)(F)C3)=O)CC2)c1 29859,Cc1ccc(C(N2CC(NC(=O)Cn3nnc(-c4cccs4)n3)C2)=O)cc1CO 29860,N1(C(c2cc(SC)oc2)=O)CCN(CC(C)NC(=O)CCCCN(C)C)CC1 29861,C1(CNC(CNC(c2c(C)occ2)=O)=O)CN(C(=O)CCCCF)CCC1C 29862,c1(C(N2CC(NC(CCS(C)=O)=O)C(O)C2)=O)cn2c(Br)cccc2n1 29863,C1(CNC(C2N(Cc3n(C)cc(Br)n3)CCOC2)=O)CCC(F)(F)CC1 29864,C1(NC(Cc2n(C)nnc2)=O)(CNC(=O)C(C)(C)NS(C)(=O)=O)CCOCC1 29865,c1(C(=O)NCC=CCNC(C2CC3CCC2CC3)=O)ccc2cc[nH]c2c1 29866,CC1OC2(C(=O)NCCC(C)(C)NC(c3cnn(C)c3Br)=O)CCC1C2 29867,N1(C(C#CC2COC2)=O)CCN(C(C2Cc3ccccc3O2)=O)CCC1C.CCS 29868,C1(C(=O)NCC2C(NC(C(C3CCCC3)OC)=O)C2)C2CCC3C(C2)CC13 29869,Cc1c(Br)c(C(N2CCC(CNC(=O)C(C)N(C)C)C23CC3)=O)nn1C 29870,C1(C(=O)NCC2CCC(NC(Cn3c(C)c(Cl)cn3)=O)C2)CCC2(CCC2)CC1 29871,C(=O)(C1=CCOCC1)N1CC(C2CN(C(CCC3(C)CC3)=O)C2)OCC1 29872,C1(CC(=O)NC(C(C)C)CNC(=O)CCN2CCCC2=O)CCCS(=O)(=O)C1 29873,c1(C(=O)NCCCCNC(CSCCOC)=O)cc(C)ccc1C1CC1 29874,c1(CC)cccnc1C(=O)NC(C)CN(C(=O)C(=Cc1ccccc1)C)CC 29875,Cc1ccc(NC(=O)COc2ccnc(F)c2F)c(I)c1 29876,N1(C(Cc2cccc(CC)c2)=O)CCC(NC(C2CC(=O)N(C)C2)=O)C(O)C1 29877,C(=O)(CC(C)(C)C#N)N1CCCC(C(C)NC(CCC(=C)C)=O)C1 29878,C1(CNC(C=Cc2c(C)nn(C)c2Cl)=O)CCC2(CC1)OCCO2 29879,n1(CC)nccc1C(=O)NC(C1CCCN1C(c1cc(CCO)on1)=O)C 29880,C12(NC(c3ccc(C)nc3)=O)COCCC1CN(C(=O)CC1CC(F)(F)C1)C2 29881,C12(C(=O)NCCc3cncc(C)n3)CC(CN(C(c3c(C)noc3N)=O)C1)C2 29882,CCCCCC(C)(C)C(=O)NCCC1(C)CCN(C(=O)CC2CCCO2)CC1 29883,Cc1c(C(=O)NCC2(C)CCCN2C(=O)C(F)(F)C(F)(F)F)nn2c1CCCC2 29884,c1(OC)ccc(C2CCN(C(=O)NC(C)C(C)(C3CC3)OC)CC2)cc1 29885,N1(C(c2nn(CC)nc2C)=O)CCC(NC(c2cc(Cl)sc2Cl)=O)C(CO)CC1 29886,N(C(=NCCCC(=O)NC(C)C)N1CCCc2ccccc2CC1)CCOC 29887,CC1(C)CC2(CC2C(=O)NCCCNC(c2cnc(C(C)(C)C)[nH]2)=O)C1 29888,C1(CNC(C2CCN2Cc2ccccc2)=O)CC(O)CN1C(C1CCC(O)C1)=O 29889,c1(OC)c(C(=O)NC(C2CCCN2C(=O)CC2(OC)CCCC2)C)ccnc1F 29890,C1(C)(C(=O)NCC(CNC(CCOc2c(C)cccc2)=O)C)CCS(=O)(=O)CC1 29891,c1(C(=O)NC(CC(C)C)CNC(=O)C(F)=CCCF)cc(Cl)ccc1C(C)C 29892,C(CCC)(C(=O)NC1CCN(C2CN(C(=O)C=Cc3cccs3)C2)CC1)=CCC 29893,Cc1cc(C(N2CCC(CF)(NC(=O)CC(C)F)C2)=O)cc([N+](=O)[O-])c1 29894,C1(C2CC2)(CNC(COc2ccn(C)n2)=O)CCN(C(C2CNC(=O)C2)=O)C1 29895,C1(C2CCC2)(C(=O)NCC(c2ccccc2F)NC(=O)CC2CCCO2)CC1 29896,C1(NC(=O)Cn2cc(C3CCC3)nn2)CN(C(C2CCC2)=O)C2(CCCC2)C1 29897,N1(C(c2cnc(C(C)=O)s2)=O)CC2(CC(NC(C3COCCC3(F)F)=O)C2)C1 29898,C#CC1CCCN(C(=O)C(C)(C)NC(C2CC3(CCC3)C2)=O)CC1 29899,C1(C(N2CC(CC=C)(NC(C3CNC(=O)N3)=O)C2)=O)CC(C)(C)CO1 29900,c1(C(=O)NCCC(C)NC(=O)C=Cc2ccc(F)cc2)cc2c(Cl)cccc2[nH]1 29901,N1(C(C(CCC)NC(N)=O)=O)Cc2[nH]nc(C(=O)N(CCC(=O)N(C)C)C)c2C1 29902,c1(CC(=O)N(C2CCN(C(=O)C3=COCC3)C2)CC)cc(C)ccc1F 29903,Cc1cc(CC(=O)N(CC(=O)N(CCC(C)C)CCO)CC(C)C)c[nH]1 29904,CC1CC(c2ccccc2)(NCC(C2CC2)NC(c2nnnn2C)=O)C1 29905,C(=O)(C(CC=C)CC=C)NC(C(=O)NCC(=O)OCC#C)CCF 29906,c1(CCC)[nH]nc(C(=O)NC2CN(C(C3CCN(C(=O)NC)C3)=O)C2)c1[N+](=O)[O-] 29907,CC1CCCN(C(=O)CC2CCCC2C)C1CNC(c1cnc(C#N)s1)=O 29908,N1(C(C(=C(C)C2CC2)F)=O)CCC2(CC1)CC2NC(c1ccc(CO)c(Cl)c1)=O 29909,C1(N(C)C(C2C3COCC23)=O)CCCN(C(=O)CSc2ncccn2)CC1 29910,c1(NC(=O)NC(C2CCCOC2)COC)ccc(C)o1 29911,C1(N(C(C(C2CCN(C(=O)CCCN3CCCC3)C2)C)=O)CCO)CCSCC1 29912,N1(C(C(c2cccnc2)C)=O)CCC(N(C(=O)C=CCF)C)CC1 29913,c1(C(N2C(C(C)NC(=O)CCc3cncnc3)CCC2)=O)c[nH]c2ncccc12 29914,Cc1cc(=NC2CCC(=O)N(C)C2)[nH]c(N2CCC(F)(CO)C2)n1 29915,C1(C(=O)NC(CCNC(CC(CC)OC)=O)(C)C)CC12CCS(=O)(=O)CC2 29916,C1(C(=O)NC)C=CC(NC(c2nnnn2CC2CCCO2)(C)COC)C1 29917,CC1CSCC1NC(C1(CNC(C2CCCCC2)=O)CC1)=O 29918,C1(CCNC(c2c(C)cc[nH]2)=O)CN(C(c2ccnn2C(F)F)=O)CC1C 29919,C(CCCC(=O)N1CCCC1(C)CNC(C1C(C(F)F)C1(C)C)=O)OCC 29920,C1(NC(c2ccc(CO)cc2)=O)CCC(NC(=O)C(F)Cc2ccccc2)CC1 29921,C1(NC(c2c(C)n[nH]c2)=O)(CO)CC2CCCC12.c12ocnc1C(=O)NOC2 29922,c1(C(N2CC3C(CNC(CC)=O)C3C2)=O)oc2ccccc2c1CS(C)(=O)=O 29923,C1(CC(=O)NC(C)CN(C)C(c2ncoc2-c2ccccc2)=O)CCCCN1C 29924,c1(C(=O)NCCCN(C(Cc2ccn(CC)n2)=O)C)cc(C(C)=O)c(C)nc1C 29925,C12(C(N(CCNC(C(CN(C)C)O)=O)C3CC3)=O)C3CCC(CC13)C2(F)F 29926,CC1CCC(CNC(c2cnc(N(C)C)cn2)=O)CN1C(=O)C=CC1CC1 29927,C1(N(C(CC=CCC)=O)C)CCCCN(C(=O)C(=Cc2ccc(Cl)cc2)C)C1 29928,C(CC(C)(C)C)(C(=O)N1CC(CNC(=O)C=C(C)Cl)C2(CC2)C1)OC 29929,C12(CCOCC1)C(=O)NC(C)C(=O)NCCO2.C(CCOC1CCC1)SC 29930,Cc1ocnc1CC(=O)NCCCC1(CNC(C2CC2C2CCCO2)=O)CCCC1 29931,c1(C(N(CC(C)NC(=O)C=C(C)C)CC)=O)ccc(OC)cn1 29932,C#Cc1cccc(C(N2CCC(CN(C)C(C3CC(=O)NC3(C)C)=O)C2)=O)c1F 29933,Cc1noc2nc(NC(=O)C(n3cc(C(C)(C)Nn4ccnc4)nn3)C)ccc12 29934,N1(C(c2n(CC)nc(Br)n2)C(=O)NC2CCC2)CCCC(C(=O)OC)(CC)C1 29935,c1(CN2CCC(CC(N3CCC(N4CCCC4)C3)=O)CC2)cccc2nonc12 29936,CCCC(CC(C)C)C(=O)NC1CC(NC(=O)CCCC(F)(F)F)CC1O 29937,C(=O)(CCCC(=O)N(CCC1(NC(C2CC3(C2)CC(O)C3)=O)CCC1)C1CC1)OC 29938,N1(C(C=CC(CC)C)=O)CCC2C(NC(c3ccc(Cl)cc3)=O)C12 29939,CCCCCC(C)CC(=O)N1CC(O)(CNC(=O)C2=NNC(=O)C2)C1 29940,Cc1noc(N)c1C(=O)NCc1cn(CC(N2CC3CC3(CN(C)C)C2)=O)nn1 29941,C(CNC(=O)C(O)CN(C)C)(CC(=O)Nc1ccccc1Cl)OC 29942,C(=O)(C(CC)C(=O)NC(C)Cn1cccn1)OCC 29943,CC1CN(C(=O)CCn2ncn(C)c2=O)CC1CNC(=O)CSCC#N 29944,Cc1cc2ccc(C(=O)NCC3(O)CCN(C(=O)Cc4ccoc4)CC3)cc2o1 29945,N1(C(c2c(C)snn2)=O)CCC(C(C)CNC(C2(P(C)(C)=O)CC2)=O)CC1 29946,N1(C(c2c(C)cns2)=O)CCC2CCN(C(c3cc4n(n3)CC(F)C4)=O)CC12 29947,c1(C(N(C)CCOCCNC(c2cccc(Cl)c2Cl)=O)=O)cccc2ncnn12 29948,c1(NC(=O)NCC2(OC)CCS(=O)(=O)C2)nccn2cccc12 29949,C1(NC(CCC(C)(C)C#N)=O)CC(NC(c2occc2F)=O)C12CCOCC2 29950,C1(C(=O)NCCCC2(NC(C(N)=O)=O)CC2)CCN2CCC1C2 29951,C1(C2(O)CN(C(=O)C(=O)NCCOC)C2)(CNC(C(CC)CCOC)=O)CC1 29952,C=C(C(=O)Nc1ccc(CCC(=O)NCC=C(C)C)cc1)C(C)(C)C 29953,CC1(C)CNC(=O)CN1c1ccn(-c2ccccc2)n1.CN 29954,Cc1ccc(-n2nc(C3CCC3)nc2CCN2CCCC(C)C2)cc1Cl 29955,O(S(=O)(=O)C=Cc1ccccc1)C1CCCN(C(COC(C)=O)=O)C1=O 29956,c1(C(=O)OC(C)C(C)(C)C)nccc2ccn(C)c12 29957,C(=O)(C(C(C)C)N(C)C)NCC(CNC(=O)Cn1nncc1C(=O)OC)OC 29958,C(CCNC(c1ccc(CC(C)C)s1)=O)(C(C)C)NC(C1(CC#C)CCCO1)=O 29959,c1(OC)cc(CC(N2CC(O)(C(C)NC(c3cnc(CC(C)C)s3)=O)C2)=O)on1 29960,N1(C(c2cc(C(C)=O)on2)=O)CCC(F)(CNC(C2(CF)CC2(F)F)=O)C1 29961,c1(C(C(=O)NCCCN(C(CCC(=C)Br)=O)CC)O)ccc(C#N)cc1 29962,C1(C(N(CCCNC(CS(=O)(=O)NCC)=O)CCO)=O)CCCC2(CCOC2)O1 29963,c1(C(CC)C)ccc(C(=O)NCC2(CNC(=O)Cn3c(C)csc3=O)CC2)cc1 29964,C(=O)(CC1=CCN(C(c2cccnc2O)=O)CC1)N(CC(C1CC1)OC)C 29965,C(=O)(C1c2c[nH]nc2CN1C(c1ccc(C(N)=O)o1)=O)N(C1C(C)COCC1)C 29966,C1(C#N)(NCc2cn(C)nc2)CCN(C(=O)C=Cc2ccc(O)cc2)C1 29967,CCC(CC(C)C)C(=O)NC1CCC(NC(=O)Cc2ccc(C#N)cc2F)CC1 29968,C(=O)(CC(O)CNC(C1CC1C(F)(F)F)=O)N(CC(CC)CC)C1CC1 29969,c1(OC)ccc(F)cc1C(=O)C(=O)NCC1CC(OC(C)(C)C)C1 29970,c1(C(=O)NC(C)C(C)C(=O)O)ccc2nc(O)nc(O)c2c1 29971,C(=O)(C(F)CC1CC1)N(C(C)CN(C(=O)CCOC1CC1)C)C 29972,Cc1cnc(C(=O)NC2CCCCC2CNc2nccc(CC#N)n2)cn1 29973,C1(C)(CNC(C2C(C(=O)OCC)C2)=O)CN(C(c2ccc(F)c(F)c2)=O)CC1C 29974,C(CC1=CCN(C(=O)Cc2cn[nH]c2)CC1)N(C1CCCN1S(C)(=O)=O)C 29975,N1(C(Cc2c(C)non2)=O)CCCC(CC(=O)NCC2CCN(C(C)C)C2)C1 29976,Cc1c(C(=O)NC(C(=O)N(CC(C2CCCC2)O)C)C(C)O)[nH]ccc1=O 29977,c1(CC)ccc(F)c(C(=O)NCC(O)CNC(c2c[nH]c(=N)o2)=O)c1 29978,C1(C(C)NC(c2[nH]nnc2C2CC2)=O)C=CC(NC(=O)CC2CCCC2)C1 29979,c1(NCCC2CCN(C(C3(COC)COC3)=O)C2)ncnc2scc(C)c12 29980,C(C(CNC(C1SCCS1)=O)S(C)(=O)=O)NC(CCNC(=O)NC)=O 29981,CC1CCCCC1OCC(=O)NCC(=O)NCCCNC(=O)Cc1csc(Cl)c1 29982,N1(C(C(C)=C(CC)C)=O)CCCN(C(C2CC3CCC(C2)C3O)=O)C(C)C1 29983,CCCC(C)(CC)C(=O)N(CCCCC(=O)NC1(C(=O)OC)CCCCC1)C 29984,c1(C(=O)Nc2ccc(OC(C)C)cc2Cl)cccc2oc(O)nc12 29985,c1(CN(C2CNC(=O)C23CC3)C=O)c(F)c(F)c(Cl)c(F)c1F 29986,c1(OC)ccc(F)cc1C(=O)N(CCC(C(C)C)NC(=O)C(F)C(C)C)C 29987,c1(C(N(CC(C)O)CCNC(C2(C(C)C)CCC2)=O)=O)cccc2c1CC(=O)N2 29988,C12(NC(c3[nH]cc(CC(C)C)c3)=O)CCCC1N(c1nnc(C)s1)CCC2 29989,C1(CCOC)(NC(COC2CCC2)=O)CCN(C(=O)C(CCSC)N(C)C)C1 29990,N1(C(C(=O)Nc2ccc(F)cc2)=O)CC2CCCC2(NC(=O)C2=CCOC2)C1 29991,n1(-c2cccc(N(CCOc3cc(C)c(Cl)cc3)C)c2)c(=O)oc2ccccc12 29992,c1(CC(CNC(C(=O)N(CC)Cc2cccnc2O)=O)CO)ccc(Br)c(F)c1 29993,c1(C(=O)NC2(CCCNC(C3(C(F)(F)F)CCCC3)=O)CC2)ccc(F)cc1N 29994,OCCC(N=c1[nH]c(=NC2CCC(F)CC2)[nH]c2ccsc12)C1CCOCC1 29995,C#Cc1ccc(C(=O)NCC2(COC)CCCN2C(C2CC2CC)=O)c(C)c1 29996,C(=O)(C(O)CC(C)C)N(CCOC)CCNC(=O)CCCc1cnn[nH]1 29997,Cc1nc(C(c2nnnn2C2CC2)NCC(C2CC2)OC)sc1C 29998,c1(OC)ccc(Cl)c(C(N2CC(NC(c3cc(O)ncn3)=O)CC(O)C2)=O)n1 29999,N1(C(CCCCCNC(C(C)C#N)=O)=O)CCc2c(C#N)cccc21 30000,C1(C(C(=O)NCCNC(C2(C(=O)OCC)CC=CC2)=O)C)CCC(C)(O)CC1 30001,N1(C(c2c(OC)nn(C)c2)=O)CCC2(NC(=O)CCc3cnn[nH]3)CC2C1 30002,n1(CC)cc(CC(=O)NCC(C)(C)NC(C2(C)CCCO2)=O)cn1 30003,c1(C(=O)NCC2(C(C)NC(CNC(CCC)=O)=O)CC2)cn(CC(F)F)cn1 30004,C1(O)(CCNC(C(=O)NCC)=O)CCN(C(=O)CCOCCN(C)C)C1 30005,C(=O)(CCCCC(N)=O)N1CCCC(CCCCNC(C(CN(C)C)O)=O)C1 30006,c1(C(N2CC(NC(C3N(C)CCC3)=O)C(C)(C)C2)=O)cnc2ccc(C#N)cn12 30007,c1(NCCCCOCCO)[nH]c(=NCc2ccc3ccsc3c2)nc2scnc12 30008,Cn1cnc2c(N3CC(CNC(c4cn(CC5CCOC5)nn4)=O)C3)ncnc12 30009,C(CCCC(C)(C)C(=O)NNC(=O)CCCCC(C)C)OCCC(C(=C)C)OC 30010,N1(C(C2CCN(C(CC3CCCC(C)O3)=O)C2)=O)CC(C)CCC12CC2 30011,N1(C(=O)COCN2CCCC2)CC(NC(C2(c3cccnc3)CC2)=O)CC1CO 30012,c1(C(=O)NCC(C(C)C)NC(=O)C(C)(C)c2ccccc2)nn(C)cc1Cl 30013,c1(C(=O)NC2CN(C(C(CC)Sc3ccccc3)=O)CC2O)cc(F)cnc1O 30014,c1(C(C)(C)C)cncc(C(=O)NCC(=O)NCCOCC(F)F)c1 30015,N1(C(C2(C)CCN(Cc3c[nH]ccc3=N)C2)=O)CCc2ccc(C#N)cc2C1 30016,C(C(C(=O)NCC1CCCO1)N(C)CC1CCCO1)(C1CCCC1)OC 30017,C(c1ccc2c(c1)COCC2)=CC(N1CCC2CN(C(c3ccsc3)=O)CC21)=O 30018,Cc1cc(C(N2CCCC(C)(NC(C3CC(CF)C3)=O)C2)=O)cc(N)c1Cl 30019,C1(NC(C2C(NC(C(C)=CC3CC3)=O)COC2)=O)CC(C)(C)C12CCC2 30020,c1(C(N(CCCNC(C2(CCC)CCC2)=O)C(C)C)=O)ncccc1Br 30021,c1(C(=O)NCC2(F)CCC(CNC(C3C(C)C3)=O)C2)n[nH]c2c1CS(=O)(=O)CC2 30022,CCC(C(C)(C)O)NC(=O)CCOCCCNC(=O)CC1CC2(CC2)C1 30023,N1(C(C2C(CCC)C2)=O)CCC(C(=O)NC2C=CCCC2CO)CC1(C)C 30024,c1(C(C(=O)NCC(C)N(C(=O)C(O)P(C)(C)=O)C)=O)cc(Cl)cc(Cl)c1 30025,c1(N(C)CC)cccc(S(=O)(=O)N(CC(C)(C)S(C)(=O)=O)CC)n1 30026,CC(C)CCC(O)C(=O)NC1CCC(CC(=O)NCC(O)CNC(N)=O)CC1 30027,C(=O)(CCC(C)(C)c1nn[nH]n1)NC(CC)C(C)C 30028,c1(CC)cc(C(N2CCC3C(CNC(c4cnsc4)=O)C3C2)=O)cn(C)c1=O 30029,C(CCCCNC(c1ncsc1C)=O)N(C(=O)CCC1CCN(C)C1)CC 30030,C(CCCC(=O)NC(COC)CC(=O)NC(C)Cc1nc[nH]n1)OCC 30031,c1(C(=O)NC2CC(OCC(=O)N(C)Cc3cc(=O)cc[nH]3)C2)ccn(C)c(=O)c1 30032,CCCCC(O)C(=O)N1CC(NCc2ccc(Br)nc2)C2(CC2)C1 30033,CC1C(C(=O)NCCN(C(C2CC(OCc3ccccc3)C2)=O)CC)CCN1C 30034,C1(F)(CNC(C2C(C(=O)OC)CC2)=O)CCC(NC(=O)CN2CCCC2=O)C1 30035,C1(CNC(CC(=O)NCC#C)=O)CC(NC(=O)CN2CCCCC2)CCO1 30036,N1(C(CCNc2ccc(C)cc2)=O)CC(CNC(c2cc(C)on2)=O)CCC1C 30037,C(c1cc(F)c(F)c(F)c1)=CC(N1CCN(C(CC(C)SC)=O)CC1CF)=O 30038,c1(OCC)ncccc1C(=O)NCCOCCCNC(=O)C(CC)n1ccnc1 30039,O=C1CS(=O)(=O)CC(C(N2CCCC(NC(=O)CSc3ccccc3O)C2)=O)N1 30040,Cn1ccc(C(=O)NC2CCC(NC(=O)CS(=O)(=O)NC3CC3)C2)c1C1CCC1 30041,C1(C(N2CC(NC(c3nc(CCC)sc3)=O)C(OC)C2)=O)CC2(CCCCO2)C1 30042,c1(C(N(CCCNC(C2(C(F)F)CCCC2)=O)C(C)C)=O)[nH]nc2ncccc12 30043,Cc1cc(F)ncc1C(=O)NC1CN(C(c2cccc(Cl)c2)=O)CC1O 30044,N1(C(C(CCC)N(C)C)=O)CCN(C(C2(C)CCC2)=O)CC1C 30045,C1(CNC2(CC(N)=O)CCC2)CC1(Br)Br 30046,CC(O)(CNC(c1cc(CCNC(=O)C(F)=CC2CC2)on1)=O)CO 30047,CCN=c1[nH]cc(CN2CCN(C(=O)CC(C(C)C)c3ccon3)CC2)s1 30048,C1(NC(C2C(OC)C2)=O)CC(NC(c2ccc(C3CC3)cc2)=O)C(O)C1 30049,c1(C(N2CCN(C(c3coc(C(F)F)c3)=O)C(CO)C2)=O)cc2cnccc2o1 30050,C1(C(C(=O)NC2CCCC2)N(C)Cc2ccc(C)o2)CC=CCC1C 30051,c1(C(=O)NC2C(NC(c3nc(COC)sc3)=O)CCC2)cnc2sc(C)c(C)n12 30052,c1(C(=O)NCCOCCOCCNC(C2C(=C)C2)=O)cc(C)c(F)c(Cl)c1 30053,C1(C)(CN(C(COCCC=C)=O)C)CCCC1NC(c1sccc1SC)=O 30054,CC(C)(C)CCC(=O)NC12CCC(NC(C3CCC(C)(C)CC3)=O)(CC1)C2 30055,N1(C(C2(C(C)C)CC2)=O)CCC2(CC1)CC(CNC(c1cc(O)ccc1F)=O)C2 30056,N1(C(c2ccsc2Cl)C(=O)NCC(C)C)CC(C)CC2CCCCC12 30057,Cc1ccc(C(N2CCC(CCC(=O)NC(C3CCCC3)CO)C2)=O)cc1 30058,n1(CCCC)nc(C)c(C(N2CCC(CC(N3CCCCC3CO)=O)C2)=O)c1C 30059,N(C(=NCCS(=O)(=O)N1CCOCC1)NCC1(C)CC1(F)F)C(COC)C 30060,c1(C=O)c(C)n(CCNC(C2(C(=O)OC)CC(CO)C2)=O)c(=O)n1C.CCO.OC 30061,C1(C(=O)NCC2CC(NC(C3COC(C)C3)=O)C2)(OC)CC(C)C1 30062,C(CNC(=O)Cn1cnccc1=O)(C(C)(C)C)NC(CN(S(C)(=O)=O)C)=O 30063,c1(C(=O)NC(CN(C(C(CSC)C)=O)CCO)C)cc2cc(O)ccc2nc1C 30064,C1(CC(=O)N(C)CCOCCCNC(=O)CC2COC(=O)C2)OCCC1(C)C 30065,N1(C(Cc2n(C)ccn2)=O)CC2CC1C2NC(=O)CC1CCC1 30066,Cc1ccc2nc(C)c(C)c(C(N3CC(C4CNCCO4)C3)=O)c2c1 30067,N1(CCCC)CCc2nc(C(=O)NCC3CCCN(C(=O)OC)C3)cn2CC1 30068,CC(=O)n1cc(-c2ccc(C(=O)Nc3ccc(O)c(C)n3)nn2)cn1 30069,CN1CC(C)(C)CC1C(N1CCC(CC(=O)NCCCN2CCCC2)C1)=O 30070,CCC(N=c1[nH]c2c(c(=NC(C)c3ncc(C)s3)[nH]1)COC2)C1CCCC1 30071,Cn1cc(C(N2CC3CC(NC(=O)COCC(F)(F)F)C3C2)=O)c2ccccc12 30072,CCC(CC)C(F)C(=O)N1CC(F)CC1CC(=O)NCc1ccc(F)c(C)c1 30073,n1(CC(=O)N(C2CC2)CC2N(C(C(C)C(C)O)=O)CCC2)ccc(=O)n(C)c1=O 30074,CCC(CC)CC(=O)N1CCC(O)(c2cn(-c3ccsc3C(=O)O)nn2)CC1 30075,c1(CC)ccc2c(c1)CCC2.c12nc(C)ccc1NC2c1nnnn1C(C)(C)C 30076,c1(OC)ccc(F)c(Cc2nc(CCC3CCC3)nn2-c2cccnc2OC)c1 30077,CCCCC(O)C(C)C(=O)NC1(C)CCCC1NC(=O)C=CC1CCC1 30078,C(=O)(C=C1SCC(=O)N1C)N1CCCC(CNC(c2c(N)cc(C)c(C)c2)=O)C1 30079,c1(C(N2CC(NC(C(C)OCC)=O)(CO)C2)=O)c(C)nc(O)nc1S 30080,C12(C(=O)NCC3CCC=CCC3)CCCC1N(C(c1sccc1F)=O)CC2 30081,Cc1ccc(C(=O)NC(C(=O)NOC2CC3CCC2C3)c2cccnc2)nc1C 30082,N#Cc1ccc(C(c2nnnn2CC(F)F)NCCC(O)c2cccs2)cn1 30083,C1(OC)CC2CC1CN(C(C1CC(O)CN1C(c1sncc1C)=O)=O)C2 30084,c12ccnc(c1)NC2=O.C1(NC(CN(C2CCC2)C)=O)(CN(C)C)CCCC1 30085,c1(COC)nccc(=NCCCCCCNC(c2csc(-c3cnc[nH]3)n2)=O)[nH]1 30086,CP(C)(=O)C(O)C(=O)NC1CCC(NC(=O)CN2CCC(O)CC2)CC1 30087,c1(C(=O)NCCCN(C(c2cc(C)c(O)nn2)=O)CCO)ccsc1S(C)(=O)=O 30088,CC(CC(=O)N1CCN(C(c2cnn(CC3CCC3)c2)=O)C(CF)C1)C(F)F 30089,N1(C(C(C)OCC#C)=O)C2CCC(C2)C1CC(=O)NCCCCCOC 30090,C1(C(N2C(COC)CC2)=O)(NC(C2CNC(=O)N2)=O)CCCC1 30091,C1(NC(=O)CC2CCOC2)C2CC1N(C(=O)C=CCO)C2 30092,Cc1cc(C(N2CC3CC(NC(c4csnc4C)=O)CC3C2)=O)c(N)c(Cl)c1 30093,C1(NC(C(CCC)C)=O)CN(C(=O)C2=CCC(C)(C)CC2)CC2(CCC2)C1 30094,N1(CCNC(C(Cc2ccco2)NC(CC2(SC)CC2)=O)=O)C(=O)CCC1=O 30095,C(=O)(CC(O)CN(C)C)NCCC(C)(C)NC(c1[nH]cc(-c2nc(C)sc2)c1)=O 30096,N=c1nc[nH]c(=NCCOC2CCN(C(=O)C=C3CCC3)CC2)[nH]1 30097,N1(C(=O)Cc2ccc(O)nc2)CC(O)C(O)C1CNC(C1(n2cccn2)CCC1)=O 30098,n1(CC)cc(CC(=O)NC2CCCC2CNC(=O)NC)cn1 30099,c1(C(=O)NCC(C)(C2CCC2)NC(CSCC)=O)ccnc2ccncc12 30100,c1(CC)ccc(F)cc1C(N1CC2CC1CN2C(C1(C(C)(F)F)CCC1)=O)=O 30101,c1(C(=O)NCC(n2cc(-c3c(COC)nns3)nn2)C)cc2n(n1)CCCO2 30102,O=S(=O)(c1sccc1I)N1CCN(S(=O)(=O)CC23CC(C2)C3)CC1 30103,Cc1nc(=N)[nH]cc1CNC(=O)NC1CCN(CC2CC2)CC1 30104,C(CC(CNC(=O)C(CO)N(C)C)NC(=O)CN(CC(C)(C)C)C)OC 30105,N1(C(=O)COCC2(CO)CNC2)CCC(c2nncs2)C1 30106,c1(C(=O)NCC(CO)NC(=O)CSc2ccncc2)cc(Br)c(Cl)s1 30107,C1(=O)CCCCCc2csc(n2)N1.N1(CC)CCC(C)CC1.C12CC1CC2=O 30108,CCC(C)C(=O)C(=O)N1CC(C)C(C)(C(N2CC(C)C(C)C2C)=O)C1 30109,N1(C(C(CO)NC(C2N(CCC)CCC2)=O)=O)CCC2(CCN(C)C2)C1 30110,C12(C(N(OC)C)=O)CC1CN(c1ccnc(NCC3CCCCO3)n1)C2 30111,c1(C(N2C(C)CC(CNC(c3ccc(F)nc3)=O)C2)=O)ccc(F)c(N)c1 30112,c1(C(=O)NC2(CNC(CCn3ccc(C)n3)=O)CC2)cn2ccc(Br)cc2n1 30113,N1(C(CCc2c[nH]c(=N)[nH]2)=O)CCC2(CC1)CC2C(N1CCC(C(F)F)CC1)=O 30114,C=CC(C)(CC)NC(c1cc(CNC(c2cocn2)=O)[nH]n1)=O 30115,N1(Cc2cc(C(=O)O)[nH]c2)CCN(C(=O)CCN2CCCCC2)CC1 30116,CC(C(C)C(=O)NCCOCCCF)NC(C1SCCS1)=O 30117,CC1CN(C(c2cn(C)cn2)=O)CC(C)C1Nc1ncnc(Cl)c1F 30118,Cc1nn2ccccc2c1C(=O)NCC(C1CC1)N(C)C(C1CCCC1(F)F)=O 30119,N(C(=NCCOC1CCCCC1)NCc1ccnn1C)Cc1cccc(C)c1 30120,c1(C(N2CCN(C(C3(C)C=CCC3)=O)CC2C2CC2)=O)ccc2ccccc2c1 30121,Cc1nc(C(F)(F)CNC(=O)NCCc2ccoc2)n[nH]1 30122,C(=O)(CCCS(N)(=O)=O)NCCCN(C(C(C)NC(COC)=O)=O)CCO 30123,C1(NC(C=CC(C)(C)SC)=O)CN(C(c2cn(C)c(=O)cn2)=O)CC2(CC2)C1 30124,c1(C(=O)NCC2(O)CCN(C(CCCCC)=O)C2)cc(OC)c(O)c(N)c1 30125,C(C)(CCC(=O)NC1CN(C(=O)CC)CC1SC)OCC 30126,c1(CN(C)C(c2cccc(CNC(=O)CCC3CC3(F)F)n2)=O)ccc(O)cc1 30127,C1(N(C(C(N2C(=O)CCC2=O)C)=O)C)CCCN(C(=O)Cn2cnnc2O)CC1 30128,Cc1ccncc1CC(N1CC2C(CNC(C3(CO)CCCO3)=O)C2C1)=O 30129,Cc1cnc(C(=O)NC(C2CCN(C(=O)C(c3ccc(F)cc3)C)C2)C)cc1Cl 30130,CC1CC(=O)NC(C(=O)NCC2(F)CCN(C(c3cnc4sccn34)=O)C2)C1 30131,CCCC(O)(CCC)CC(=O)NC1CC2CC(C1)N(C(c1c[nH]c(=O)cn1)=O)C2 30132,C1(NC(C2CCCCC2(F)F)=O)CC2CC(NC(=O)CC3=CCOCC3)CC2C1 30133,N1(C(c2ncc(C)c(C)c2)=O)CCC2(C=C(C(=O)N3CC(CO)C(O)C3)C2)C1 30134,N1(C(c2cc(C)ncc2)=O)CCC2CCN(C(=O)C(CN(C)C)N(C)C)CC12 30135,n1(CC(=O)NCC23CC4CC(CC(C4)C2)C3)ccc(=NC(=O)C#CC2CC2)nc1O 30136,Cc1cnn(CCC(=O)NCCOC2CN(C(C3CCCN3C)=O)C2)c1 30137,C(=O)(C(CC(C)C)NC(c1cccs1)=O)NCC(CC)NC(=O)CC1CN(C)C1 30138,c1(CCC)onc(C)c1C(=O)NCCCN(C(=O)C=CC(CC)=CC)C 30139,c1(C(N2CCC(NC(C)=O)C2)=O)cc(CNC(C2COCC(C)O2)=O)nn1C 30140,C(=O)(C(C)(C)C#N)NCC(C)(C)CC1CN(C(c2ccsn2)=O)C1 30141,C(C(O)C(=O)N(CC(C)C(=O)NCC1CSCCO1)C)SC 30142,C(C(=O)NC(CO)C(C)NC(C1(CCF)CCC1)=O)(C(C)C)SCC 30143,S(=O)(=O)(c1cccc(C(=O)N=c2cc[nH]cc2Cl)c1)NC(COC)COC 30144,N1(c2ccnc(C)n2)CC23CCCCC2(CN(C(C2(CC4CC4)CC2)=O)C3)C1 30145,N(C1CCc2sc3c(c21)CCCC3)C(c1cn(CCN(C)C)nc1)=O 30146,c1(C(N(CC(CNC(Cc2cc(C)nn2C)=O)(C)C)C)=O)cc2n(c1)CCSC2 30147,C=C1CCN(C(=O)CC=CCC)C(C(N2CCC(CF)CC2)=O)C1 30148,c1(CCNC(C(CC)N(C)C(c2cc(C3CC3)[nH]n2)=O)=O)noc(=O)n1C 30149,C1(CC(=O)NCCC2(NC(C(C(C)C)C)=O)CCCC2)COC(C)(C)CO1 30150,c1(C(=O)NCCC2(O)CCN(C(=O)C3=CCSC3)CC2)cc2c(nn1)CCC2 30151,C1(C(=O)OC)(C(=O)NC2CCCC2CC(=O)NCC2(COC)CC2)CCOC1 30152,C(=O)(C(C)S(=O)(=O)C(C)C)N1CCC(OCCCNC(C(COC)(F)F)=O)CC1 30153,CCC(C)C(=O)C(=O)N(C)CC1(O)CCCN(C(c2sccc2CO)=O)C1 30154,Cc1cc(F)c(CNC2CN(C(=O)Nc3cccc(Br)c3)CCC2F)c(Br)c1 30155,N1(C(CC(C)CN(C)C)=O)CCCC(CC(=O)NCCN2CC3CC3C2)CC1 30156,C1(C(N(CCN=[N+]=[N-])CC)=O)CCOCC1NC(C1(C)CCN(C)C1)=O 30157,N1(C(C=Cc2c(C)nccc2)=O)CC(C2CCCCN(C(=O)CSC(F)F)C2)C1 30158,C(C1=NOC2OCCC12)NC1C(CN)CCC=C1 30159,C1(C(=O)NC(CC#C)CCOC)CCN(C(=O)c2csc(C)c2)O1 30160,N1(C(C(C)OC)C)CCC(O)(C(=O)N(CCCN(C)C)C)CC1 30161,N1(C(CCC#N)=O)CCCCC(N2CCC(OCC(F)(F)F)C2)C1=O 30162,C1(OCC)CCCC1OC(=O)C(c1ccnn1C)C 30163,CCCC(CC(=O)N1CCC1CC1CC1)c1ccccc1.n12nnnc1CC2=O 30164,C(=O)(CCC(=O)N1CCOC(C2CN(C(c3coc(C)c3)=O)C2)C1)OC 30165,c1(C(=O)NCCCN2CCN(C(C3(O)CC3)=O)CC2)cc([N+](=O)[O-])ccc1Br 30166,N1(C(=O)C2=COCCO2)CCCN(C(c2cc[nH]c3nccc2-3)=O)C(CO)C1 30167,C1(C(N2C3CN(C(c4ccc(C)nc4)=O)C(C3)CC2)=O)CCc2ncccc2C1 30168,Cc1ccc2c(CC(=O)NC3CC(NC(C4(CO)CCCCC4)=O)C3)coc2c1 30169,N1(C(c2cccnc2S)=O)CCC2(CCCN2C(c2ccc[n+]([O-])c2)=O)C1 30170,c1(CN(C(c2ccc(C(=O)OC)n2C)C(=O)NC2CC2)C)c(C)nn(CCl)c1C 30171,C1(C(=O)Nc2cnc[nH]2)CN(Cc2ccc(Br)cc2)CCC1O 30172,N1(C(C2C(NC(CCCN=[N+]=[N-])=O)C=CCC2)=O)CCC12CCCCC2 30173,c1(C(N2C(CO)CC(NC(C=C(C)C)=O)C2)=O)cc2c(Br)coc2cn1 30174,N1(C(c2c(CC)nn[nH]2)=O)CCC2(CCCN2C(=O)CCCC2OCCO2)C1 30175,c1(C(N2CCC(O)(CNC(C(n3c(C)ncc3)C)=O)C2)=O)nnn2c1CCCC2 30176,Cc1cccc(N2CCC(NC(C3CCC(N4CCOCC4)C3)=O)C2=O)c1 30177,C(=O)(CCCCCN(C)C)N(CC(CC)NC(=O)CSc1n[nH]c(C)n1)C 30178,C1(NC(c2c(C(=O)OC)[nH]cc2)=O)CCC(NC(=O)COCC(F)(F)F)CC1 30179,Cc1cc(C(N2CC3CCC2C(NC(C2CCC2)=O)C3)=O)c(N)c(F)c1 30180,C1(NC(Cc2c(C)ccs2)=O)CN(C(C2(C(=O)N(C)C(C)C)CC2)=O)CC1C1CC1 30181,CC(C)CC(C)C(=O)N(CC(O)CNC(=O)COc1ccc(CC#N)cc1)C 30182,c1(C(N2CC(NC(C34CCN(CC3)CC4)=O)C2)=O)ccc([N+](=O)[O-])[nH]1 30183,c1(C(=O)NC2C(CNC(CN(CCC#C)C)=O)C2)ncccc1OC 30184,C(CC1=CCN(C(c2ccc(C)c(C(=O)OC)c2)=O)CC1)NC(CCC=CC)=O 30185,N1(CC(N2CC(C(=O)N(CC(=O)O)CCO)CC(C)C2)=O)CCc2ccccc21 30186,N1(C(c2c(C)coc2)=O)CC(NC(c2[nH]nnc2C)=O)CC1C 30187,C#CCCCC(=O)N(CC(N1CCN(C(C2CC(O)C2)=O)CC1)=O)C 30188,C1(NC(CCC=C=C)=O)CC=C(C(=O)N2CCC(OC(C)=O)C2)C1 30189,Cc1cccc(F)c1C(=O)NC1CCC(NC(C2CC23CC3)=O)CC1 30190,N1(C(C(C)(C)c2cccs2)=O)CCCC(O)(CNC(c2ccc(C(F)F)o2)=O)C1 30191,CCC(CC(=O)NOCC(=O)NCc1nccs1)C(C)(C)C 30192,N1(C(CCOCCOC)=O)CCC(C(=O)NC(CCO)C2CCC2)(CC)CC1 30193,n1(CC(N2C(C)CC(CNC(=O)CC3CS(=O)(=O)C3)C2)=O)nnc2c1CCCC2 30194,c1(C(=O)Nc2ccc(C#N)cc2)cnc2c(-c3ccc(CO)nc3)cccc2c1 30195,CCCCC(CC)C(=O)NCC(C)(F)CNC(c1ccn(CC)c1C)=O 30196,c1(C(N2CC(NC(c3ccccn3)=O)C3C2C3)=O)ccc2cnccc2n1 30197,C1(C)(NC(CCCN(C)C)=O)CCN(C(=O)C2=CCCC2)CC1 30198,N1(CC)CCCCC1C(=O)NCCC1(NC(c2cnn(CC(F)(F)F)c2)=O)CC1 30199,N1(C(=O)OC(C)(C)C)C2CCC1CC(CNC1CCC(O)CC1)C2 30200,C(=O)(C(CN(C)C)C(C)C)NCC(C)(C1CCC1)NC(Cc1cc(C)n(C)n1)=O 30201,C1(C(=O)NC(CC=CC)C(=O)N(C)CC2(F)CCCC2)C2CCC(C2)C1C 30202,c1(-c2n(C)cnc2)ccc2oc(C(=O)Nc3cc(O)ccc3Br)cc2c1 30203,c1(C(=O)OCC)cnc(NC2CC(C)N(C(C3CC4(CCCO4)C3)=O)C2)nc1C 30204,C(C(=O)NCCOCc1cccc(Cl)c1)(C(C)CC(C)C)N(CCCSC)C 30205,c1(C(=O)NCC(CC)NC(=O)C(CC)Nc2nc(C)cs2)cccc(=O)o1 30206,Cc1c(C(=O)NCC2CC3C=CC2C3)cc(Br)cc1Cl 30207,CC(F)(F)C(C)(C)CNC(C1(NC(=O)COCC2CCCO2)CSC1)=O 30208,N1(CC(=O)NCC(O)CNC(c2csnn2)=O)CCCC1CO 30209,Cc1cc(C(=O)NC2CC23CCN(C(=O)COCC(F)(F)F)C3)nc2nccn12 30210,CN1CCOC(C(=O)N(C)C(C2(F)CCC(NC3(c4cc[nH]n4)CC3)C2)=O)C1=O 30211,c1(OC)ccc2c(C(N3CCC(Nc4c([N+](=O)[O-])c(C)nn4C)C3)=O)cnn2c1 30212,C1(CC)CCCC(C(N2CCCCC2CCN2CCCC2)C(=O)NC(C)(C)C)C1 30213,N1(CC(N2CC(O)(CCNC(CCCOCC)=O)C2)=O)OC(C)(C)CC1=O 30214,C#CCCCCCC(=O)N1CCCOC(CNC(=O)Cn2cccc2)C1 30215,C1(NC(c2cc(O)nc(O)n2)=O)COC2(CCN(C(c3cccnc3Cl)=O)C2)C1 30216,CC1CN(C(=O)CC(C)(C)CCC2OCCO2)CCC(c2nc(C3CC3)no2)O1 30217,c1(NC2(CC(=O)NCC(N3CCCS3(=O)=O)(C)C)COC2)ncc(C#N)cc1Br 30218,c1(C(=O)NC2(C)CC(NC(CC3(C)CCCO3)=O)C2)ccc(CO)cc1F 30219,Cc1ccnc(CNc2c[nH]nc2C(=O)Nc2nccnc2C(F)(F)F)c1 30220,C1(CCNC(C2(CC#C)CC2)=O)CCCN1C(=O)COC(C)CC 30221,c1(N(C2CCCN(C(C3CC3CC)=O)C2C)C2CCC2)cc(OC)c2c(c1)CCO2 30222,N1(C(CCNC(C(C=C)C)=O)=O)CC=CCC1C(=O)NC 30223,N1(C(C2(C=C)CCN(C(=O)CC(C)SC)C2)=O)Cc2cccc(O)c2C1 30224,n1(CC)ncc(C(=O)NCC2CCN2C(c2ccc(C)s2)=O)c1C 30225,CCC(CNC(C1(n2ccnn2)CC1)=O)NC(=O)Cc1cnc[nH]1 30226,c1(C(C)C)cc(C(=O)NCCCOCCOCCNC(C2C(C)C2C)=O)on1 30227,C=CCC(C)(CO)CN=c1[nH]c(=NCc2nc(C(C)C)ns2)[nH]c2c1COC2 30228,c1(CC(=O)NCC2(C)CCN(C(Cn3nnc(C)n3)=O)C2)c(F)cncc1Cl 30229,Cc1ccc(OCC(=O)NC(C)(CNC(c2cn(C)cn2)=O)C2CCC2)cc1C 30230,Cc1c(C(N2CC(NC(C34CC(C(C)C)(CO3)C4)=O)C2)=O)[nH]c2ccccc12 30231,c1(C(C(=O)NC(CSC)CC(C)C)C)c(Cl)cccc1Cl 30232,N1(C(CN2CC(C)(OC)C2)=O)CCN(C(=O)C2=CCCN(C)C2)CC2CCCCC12 30233,S(=O)(=O)(CCC(=O)NCC1CC(C(F)(F)F)CN1Cc1cccc(=O)n1C)NC 30234,c1(C(=O)NC(CC)CNC(=O)CN2CCN(C)CC2)cnc2ccccn12 30235,N1(C(c2c(C)oc(C(C)C)n2)=O)C2CCC1CC(N(C(=O)C(C)CC1CC1)C)C2 30236,C1(C(=O)OC)CNC(=O)CC12CCN(C(=O)CCCOc1cccc(Br)c1)CC2 30237,C=CC1OCCC1N=c1[nH]c(N2CCN(CC(F)(F)F)CC2)nc2ccccc12 30238,N1(C(C2N(C(=O)C3=CCCCC3)CCN(C)C2)=O)CCn2ncc(O)c2C1 30239,C12(C(N(C(CNC(CC(C=C)C)=O)C)CC)=O)C3CC(CC13)C2(F)F 30240,C1(C(C)O)CCN(CCN(c2cc(Br)n(C)n2)C(=O)C2CC2)CC1 30241,N1(C(c2n(CC)ncc2)=O)CCCC(C)(C(=O)NCCNC(=O)OC)C1 30242,CCC(C)CCC(O)CC(=O)N1CCC(NC(C2CC(=O)C2(C)C)=O)CC1C 30243,CC1CCN(C(C2COC(=O)N2C)=O)CC1NC(=O)C(C)(C)F 30244,O(NC(=O)C(C)(C)C#C)CC(=O)NC(C#C)C(C)C 30245,Cc1cccn2cc(C(N3CC(CNC(C4C(C#N)C4(C)C)=O)CC3C)=O)nc12 30246,C1(CC(=O)NCC2(NC(=O)CSc3ccc(F)cc3)CCOC2)CCCC12CC2 30247,c1(C(N2CCC(C)(C(=O)Nc3cc(Cl)ccc3CO)C2)=O)cc(F)c(Cl)cc1O 30248,c1(C(=O)NCC2C(NC(Cn3ccc(C)cc3=O)=O)C2)c(C)cc(C)nc1O 30249,c1(CC)nn(C)c(CC)c1C(=O)NCCC(C)N(c1cc(Cl)c(O)nn1)C 30250,c1(C(=O)NC(C(CC)C)C(N2CCC3(CC(CO)C3)C2)=O)ccn2nccc2c1 30251,c1(C(=O)NCC(C)(C2CC2)NC(C(C)OCCCC)=O)cc(O)cc(C#N)c1 30252,C1(CNC(C2(C)CCC(=O)C2)=O)CC(C(=O)NC2(CC(N)=O)CC2)=NO1 30253,N1(C(Cc2c(C)nc(Cl)cc2)=O)CC2CN(C(=O)Cc3ccc(F)cn3)CC2C1 30254,C(C(CC1CCCC1)C(=O)NOC1CCOC1)NC(CC1(CC)CCC1)=O 30255,C1(C(=O)NC(C2CCN(C(C3(n4ccnn4)CC3)=O)C2)C)CCCCC(F)(F)C1 30256,CCC(C(=O)NCCOCCOCCNC(C1CC2CC1C2)=O)C(C)C 30257,N1(C(CC(C)(C)C#N)=O)CCC(O)(C2CCN(C(C3CC(=O)N(O)C3)=O)CC2)C1 30258,C1(C2CC2)(CNC(CC2C(C)=NNC2=O)=O)CCOCC1 30259,c1(C(N)=O)ncn(CC(=O)NCC2CCC(NC(C3CC4CC4C3)=O)C2)n1 30260,N1(CCCC(=O)NCCN(C(=O)CC(F)F)CCC)C(=O)NC(C)(C)C1=O 30261,c1(C(N2CCCN(CCOC)CC2)C(=O)NCCSC)ccc2c(c1)CCCS2 30262,C1(C)(N)CCN(C(C)=O)C1.C(CCC=O)OC.C1(C(C)C)CNC(=O)N1 30263,c1(NC(C2CC(NCc3ccc(CO)cc3)C2)=O)ccc2sncc2c1 30264,Cc1cn(C)nc1C(=O)N(CC(C)CNC(C1CCCN1S(C)(=O)=O)=O)C 30265,c1(NCC(CC)(C)C(C)O)nc2ccccc2nc1NCCN1CC2CC2C1 30266,CC1C(NC(=O)COC2CCOC2)CCN1C(=O)C=CC1CCC1 30267,N1(C(c2scc(C)c2)=O)CCC2(CC1)CC(C(N1CCCC(C)(F)CC1)=O)C2 30268,C=C(C)C(C)(C)C(=O)NC1CCC(N(C)C(c2ccccc2C(C)O)=O)CC1 30269,S(=O)(=O)(c1ccccc1F)NC(C1C(NC(c2cccc(F)n2)=O)C2CCC1C2)=O 30270,N(C(=NCCc1ccns1)NCC1CCC(C)(C)C1)Cc1ccc(OC)cc1 30271,CC1CN(C(=O)COC2CC2)CCCN1C(=O)CC12CCC(CC1)OC2 30272,CC1OCCC1C(=O)NCC1CCOC1C(=O)NCCc1cnn[nH]1 30273,C1(CNC(=O)NC)CCN(C(=O)Cn2ccnc2C(C)C)CC1 30274,C(C(C)(C)C(=O)N1CCCCC1Cn1cc(C2(O)CCC2)nn1)OC 30275,Cc1sc(=O)n(CC(=O)NC(C2CCCN2C(c2cc(Cl)ccn2)=O)C)c1C 30276,C(C)(CO)(C(=O)NC1(CCF)CC(O)C1)NC(CC(C)n1cccn1)=O 30277,C=C(Cl)CC(C(=O)N=c1cc(C)n(CCO)[nH]1)NC(=O)C1=CC2(CCOC2)C1 30278,C(=O)(C1=NOC2(CCOC2)C1)NCCOCCNC(C1(c2c(C)c[nH]n2)CC1)=O 30279,CC1C(=O)N(CC(=O)NCCCN(C)C(c2nc(=N)cc[nH]2)=O)C(=O)C1C 30280,C1(C(=O)NCCC2CCN(C(C(C)=C3CCCC3)=O)CC2)CC(F)(F)C12CCC2 30281,C(C(=O)N=c1ccn(CC(C)C)[nH]1)N(C1CN(C)CCO1)CCC 30282,N1(C(CCC(C)OC)=O)CCC2(CCC(NC(=O)CCc3ccoc3)C2)C1 30283,C1(C(=O)NC23CC(NC(C4(CN(C)C)CC4)=O)(C2)C3)CCC(N(C)C)CC1 30284,C1(CNC(C23CC(C4COC4)(C2)C3)=O)CC(CNC(C2CCC2(F)F)=O)CO1 30285,C(=O)(C1CCCc2scnc21)NCC(C)(Cn1cccn1)NC(C(=O)NCC)=O 30286,C1(NC(c2cc(CC)ncn2)=O)CN(C(=O)C(=O)C(C)CC)CC(F)(F)C1 30287,C(=O)(C#CC1CCCC1)NCCCN(C(=O)CCN1CCSC(C)(C)C1)C(C)C 30288,C(CCC(C)C)(C(=O)N1CCC(F)(CO)CC1)NC(C(=CC1CCCC1)C)=O 30289,C1(CC(=O)NC2(CNC(=O)CC3CCCCC3)CCOC2)CCCS1(=O)=O 30290,C(=O)(C(F)C(C)CNC(=O)C=C1CCCCC1)N(C(C)C(=O)OC)CC 30291,c1(C(N(C(C)C)CCNC(=O)CN2CCNC(=O)C2)=O)n[nH]c2ccc(F)cc12 30292,N1(C(c2ncn(C)n2)=O)CCOC2CN(C(=O)CC3CCC(C)(C)O3)CC12 30293,c1(C(=O)NCCC2(C(=O)NC(c3ccncn3)C)CCC2)ncccc1N 30294,N1(CCC)CC(C(=O)N(CCCCCNC(=O)COCC(C)(C)C)C)CC1=O 30295,S(=O)(=O)(c1ccc(C#N)c(N2CCC3CC3C2)c1)N1CCCC(=C)C1 30296,c1(C(C)C)ncc(Cl)c(C(=O)NCCC(C)NC(=O)Cc2cnns2)n1 30297,C12COC3(CC1C3)C(=O)N2.c1(OC)ccc(C(=O)N(C2CCCC2)C(C)C)cc1 30298,c1(N2C(=O)CN2CC(C)C)cccc(Cl)c1F.c1(CC)nn[nH]c1C(=O)O 30299,c1(C(=O)NC2(C)CC(NC(Cn3c(C)nnn3)=O)C2)cccc2c1OCC2(C)C 30300,CC(C)CC(C(=O)NC1CC2CC(NC(=O)CSc3nnnn3C)C1C2)C(N)=O 30301,C(=O)(C1C(=O)N1)OCC.C(=O)(CCSC1CC1)N(C(C)CCOCC)C1CC1 30302,C1(CC)CCC(C(=O)ON2CCC(O)(c3ccc(C)nc3)C2)CC1 30303,N1(C(C(CC(F)F)N(C(CNC(=O)NC)=O)C)=O)CC2(CNC(=O)N2C)C1 30304,c1(OC)ccc2nc(N3CCC(NC(=O)Cn4cc(C(C)O)nn4)C3)sc2c1 30305,N1(C(c2ccc(N(C)C)cn2)=O)CC2(CCCN(C(c3cc(O)nn3C)=O)C2)C1 30306,C1(COC)CN(C(=O)Cc2cncc(Br)c2)CCN1C(=O)CC(C)OC 30307,C(C(CC(C)C)C(=O)NC(C)(C)CNC(C1(C)CC1)=O)OC 30308,c1(N2CCC(CC)C2)ncc(C)cc1S(=O)(=O)N1CCC1(C)NC(=O)NC 30309,C(=O)(C1=CC(O)CCC1)N1C(CN(C(=O)CCCC2CCOCC2)C)COCC1 30310,Cc1ccc(C(=O)NCC(=O)NC(C)CCNC(=O)CCC(C)C)cc1C 30311,N1(C(c2c(C)nsc2C)=O)CC2(CO)CC1(C(=O)NCC1(C)CC1(C)C)C2 30312,N1(C(c2c(C#N)nc[nH]2)=O)CC2CCC2(CCNC(=O)C(=O)NCC(F)F)C1 30313,C1(NC(C2CC(C#C)(O)C2)=O)CS(=O)(=O)CC1NC(=O)C=C1CCN(C)CC1 30314,C1(C(=O)NCCC(N2CCCCC2)C)CC2CCC(N2)C1C(F)(F)F 30315,CC(C)CC(O)CC(=O)N1CCC=CC1C(=O)NCC1(C)CC1(F)F 30316,C1(CNC(C2CCOC2)=O)CC2COCC2N1C(=O)CCc1ccc(Cl)nc1 30317,N1(C(C)C)C(=O)CCC1C(=O)NC(C)(CNC(c1c[nH]c(=N)o1)=O)C1CC1 30318,CC1c2ccc(Br)c(Cl)c2CCN1CC(c1c(F)cccc1F)=O 30319,CC1=C(C(=O)NCC2C=CC(NC(=O)CC3CCC3)C2)C(C)n2nnnc2N1C 30320,C(=O)(CC(CC)C(C)(C)C)N(C1CCN(C(c2nc(C)c(C)[nH]2)=O)C1)CC#C 30321,C(=O)(C1=CCC(C)CC1)NCC(CC=C)NC(c1ncsc1S(N)(=O)=O)=O 30322,c1(C(N2CCC(C(C(=O)Nc3c(CC)cccc3)C)C2)=O)ccc2cncn2c1 30323,C1(CNC(Cn2c(CCC)ncc2)=O)CC(F)CN1C(c1cnncc1OC)=O 30324,C(=O)(CC(F)(F)C(F)F)N1CC(NC(=O)C=Cc2ccsc2)C(F)C1 30325,c1(C(=O)NC2C(OC)COC2)ccnc(CNC(=O)C(C)(C)NC(C)=O)c1 30326,C#CCCCCCC(=O)N1CCC(NC(c2c(C)cccc2Cl)=O)CC1C1CC1 30327,c1(CC(=O)NCCC2CN(C(=O)N(C3CCC3)C3CC3)CCO2)cccc(I)c1 30328,N1CC(NCc2scc(OC)c2)CC1(C)C.C1(=O)CC(C)(C)O1.c1ccccc1 30329,c1(CC)nn(C)c(CC(=O)NCC2COCCN2C(c2ccnc(O)c2)=O)c1Cl 30330,N1(C(c2cc(C)c(C)s2)=O)CCCC(O)(CN(C)C(C2(C)CC(C)(C)C2)=O)C1 30331,c1(CC(=O)NCC(CC=C)NC(c2ncc(C)cc2C)=O)csc2ccccc12 30332,Cc1cccc2c1c(CN1CCC(C#N)(NC(=O)C(C)n3cccn3)C1)cn2C 30333,C1(C(=O)NCC2CN(C(=O)CC3CCCCO3)C2)(COC)CCCCO1 30334,C1(NC(=O)CC(O)c2cnc(Cl)s2)CN(C(c2cnco2)=O)CC12CC2 30335,N1(C(CC2C(C)=NNC2=O)=O)CCCCC(CCC(=O)N(C)CC2CC2C)C1 30336,C1(CCCCNC(c2c(C)c[nH]n2)=O)CCN(C(c2c[nH]ccc2=O)=O)CC1 30337,C=C=CCCC(=O)NC1(CCNC(=O)CC2(OOc3ccccc3)CC2)CCC1 30338,CN1CCC2CN(C(C3CC(NC(C4(O)CCC4)=O)C3)=O)CC2C1 30339,N1(C(C2CCC(OC)CC2)=O)C2CC1CN(C(C1(C)CNC(=O)C1)=O)C2 30340,N1(C(C2C=CCN(C(C3CCCC(OC)C3)=O)C2)=O)CCC(C2=NOCC2)C1 30341,C1(NC(CCCOC)=O)CC=C(C(=O)NC2(C(C)O)CC2)C1 30342,C1(C(N(C(C)C(N2CCC(CN=[N+]=[N-])C2)=O)CC)=O)CCOC1(C)C 30343,n1(CCC)cc(C(=O)N(CCC(=O)N(C2CCCC2C)C)CC)nn1 30344,C1(NC(c2c(N)cncc2)=O)CC(NC(c2cc(C(F)F)cs2)=O)C12CCC2 30345,N1(C(CCC)C)CC(C(=O)NC(C)CNC(C2(C(F)F)CCCC2)=O)CC1=O 30346,CC1C(C=CC(N2CCCCC2CCNC(c2cscn2)=O)=O)C1(Cl)Cl 30347,Cc1cccc2cc(C(=O)NC3CCCC3NC(=O)C#CC3CC3)[nH]c12 30348,N1(C(c2ccc(OC)c(OC)n2)=O)C2CCC1CC(N(C)C(C1OCCO1)=O)C2 30349,c1(NC(c2cn(Cc3cccnc3)nn2)=O)cccc(O)c1 30350,c1(C(=O)NC(CC(C)NC(c2c(C)nncc2)=O)C)ncc(C#N)cc1Cl 30351,CC12COC(C(=O)NCCC3CSCCN3C(=O)CC3CCCCC3O)(C1)C2 30352,c1(NC(C2CCS(=O)(=O)C2)=O)cccc(-c2ccccn2)c1Cl 30353,Cc1cc(C(=O)NC2CC(CNC(c3cccc(Cl)c3C)=O)C2(C)C)cc(O)n1 30354,Cc1cnc(F)cc1NC(=O)CN(C)C(=O)OC(C)(C)C.c12ccc(cc1)s2 30355,N1(C(CCC=C)=O)CCC(C)(C(N2CCC(C)(C(C)C)C2)=O)C1 30356,C1(C(=O)NC(CC#C)C(=O)NCc2nc(C(C)C)n[nH]2)CC2(CCO1)CC2 30357,c1(N(C)C)ccccc1NC(C1C=CC(NCc2csc(Br)c2)C1)=O 30358,C(=O)(CCC(=O)NN(C)C)NC(C1C(C(=O)NCC(CCC)C)C1)C 30359,C1(CCOC)(NC(=O)C(C)N(C)C)CCN(C(C23CSC(C2)C3)=O)CC1 30360,n1(C(C)C)nnnc1C(C1C=CCC1)NCCCN(S(C)(=O)=O)C 30361,C1(NC(c2c(CC)nc(C)n2C)=O)CCN(C(=O)Cc2cncn2C)CC1(C)C 30362,N1(C(CCCC(C)C)C(=O)NC(C)C)CCc2ccc(F)c(F)c2C1 30363,N1(C(c2ccc(Oc3ccccc3)o2)C(=O)NC)CC2CCC1CN2CC 30364,Cc1ccc(F)cc1C(=O)NC1CCCN(C(=O)Cn2ccc(C(F)(F)F)n2)C1 30365,C(=O)(C(C)(C)C(C)O)NCc1cccc(CN(C(CC(C)O)=O)C)c1 30366,N1(C(C(CC)N(C)C)=O)CCCC2(CC(NC(=O)C(C)OCCC(C)C)C2)C1 30367,CCC(COC)C(=O)NC(C)CNC(c1cc(Cl)cnn1)=O 30368,CCCCCC(O)CC(=O)NCCC1CCCCN1C(=O)C(CC)SC 30369,C1(NC(c2ncnc(=N)[nH]2)=O)CC2CC(NC(c3ccno3)=O)CC12 30370,C1(C(CC)C)CCN(c2cc(N3CCOC(c4nncn4C)C3)ncn2)CC1 30371,C#CC1(C)CCCN(C(=O)C(CC(=C)C)NC(c2cc(C3CC3)[nH]n2)=O)C1 30372,C1(CNC(c2[nH]cc(C)c2)=O)COCCN(C(c2nc(CC(F)(F)F)cs2)=O)C1 30373,C(=O)(C(C)(C)CCSC)NCC1CC(COC)CN1C(=O)CNC(=O)C1CC1 30374,CC(C)N(NC(=O)C1CCCCO1)C(=O)Nc1nccs1 30375,c1(CC)ccc2c(c1)CN(c1nnc(-c3ncc[nH]3)n1CCC#N)CC2 30376,c1(OC)nn(C)cc1NC(c1ccc(CNC(=O)C(O)CC2CCCC2)cc1)=O 30377,Cc1ncc(C(=O)NC(C2CCCCC2)CNC(C2(CF)CCOCC2)=O)c(C)n1 30378,Cc1cccnc1C(=O)NC(C1CCCN1C(c1ccsc1)=O)C 30379,c1(C(N2CCC2CF)=O)ccc(-n2cc(-c3c[nH]nc3F)nn2)cc1 30380,N1(C(c2cnc(CC)s2)=O)CCCCC(N(C(=O)C(O)CC2CCOCC2)C)C1 30381,c1(C(N2CC(NC(C(C)n3ccnc3)=O)C(C)(C)C2)=O)c(O)cc(Cl)cc1F 30382,C1(NC(C2(CCOC)CC2)=O)CCCCC1CNC(=O)Cc1ccncc1 30383,c1(CNC2C(F)CCN(C(C3CC4C=CC3C4)=O)C2)cc(C(F)(F)F)ccc1Cl 30384,C(=O)(CCCCC(=O)N(C)CCNC(=O)Cn1cc(Br)c(C)n1)OC 30385,c1(OC)ccc2cccnc2c1C(N1CCC(CNC(=O)C(C)C#N)C1)=O 30386,N1(C(C(CO)N(C)C)=O)C2CCC1CN(C(c1cccc(C(C)(C)C)c1)=O)C2 30387,c1(C(=O)OC)cc(Cl)nc(Cl)c1NC(C1(C)CCN1Cc1cscn1)=O 30388,c1(C(N2CCCC2CCNC(C23C=CC(CC2)C3)=O)=O)ccc2c(c1)COC2=O 30389,C(=O)(CCCC(=O)N(C)C)N1CC(OC)C(NC(c2cnn(C(C)C)c2Cl)=O)C1 30390,N1(c2nnc(C(CC)(C)C)o2)CCCC(C)(NC(=O)C(C)=C(C)C)C1 30391,C1(C(=O)NCC2CC3(CC3)CN2C(c2ccc[nH]2)=O)CCC(C2CC2)CC1 30392,C1(C(=O)OCCn2nccc2N)(CNC(=O)OC(C)(C)C)CCCO1 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30411,C(C1=CCN(C(C2CCC(CCO)CC2)=O)CC1)NC(c1cn(C)nn1)=O 30412,Cc1cc(C(=O)NCC2C(CNC(c3cc(C)oc3C)=O)C2(F)F)c(C)[nH]1 30413,CC(C)(C(=O)NC1CC(F)(CNC(c2cc(C3(C)CC3)on2)=O)C1)C(N)=O 30414,c1(CCC(=O)NCC2(CN(C(CCSC)=O)C)CC2)ccc(Cl)cc1 30415,c1(C(N2CCC(OCCNc3snc(COC)n3)C2)=O)cnc(C(F)(F)F)cn1 30416,C(=O)(C1=NOC(C)C1C)N1CCC(C(C(=O)NCCC(=O)NC)F)C1 30417,CC1C(C(N2CCN(CC3(NC(C4(C)CCCN4C)=O)CC3)CC2)=O)CCN1C 30418,c1(CC)nc(CC(=O)NCC2CCN(C(=O)CSC3CCCCO3)C2)cs1 30419,C1(C(=O)NC2(CNC(CNS(C)(=O)=O)=O)CC2)CC12CCC1(CC1)CC2 30420,c1(C(=O)NCc2c(C(=O)NC(C=C)C3CC3)nco2)cccc(Cl)c1 30421,c1(C(=O)NC(CNC(CCOCC)=O)(C)C2CC2)ccc(C2(C#N)CC2)cc1 30422,c1(C(N2CC(CNC(COC)=O)N(C)CC2)=O)cc2ccccc2n1CC(F)(F)F 30423,c1(SC2ON=C(C)C2)cccc(CC(=O)N(C)Cc2ccccc2)c1 30424,C1(NC(C(CCC)C)=O)CCC12CN(C(=O)CCCCN1CCCCC1)C2 30425,c12cc3ccc(cc3o1)NC2=O.C(=O)(CCC(C(=O)O)NC(C)=O)OC 30426,C(=O)(C(C)Cc1cn(Cc2cn(C(C)C(=O)O)nn2)nn1)N(C1CSC1)CC 30427,CCC(C)C(C(=O)NC1CCCCC1C(N1CC=CC1(C)COC)=O)N(C)C 30428,c1(C(N(C2C3CN(C(=O)CC4(C)CC4)CC23)C)=O)ccc(Cl)cc1 30429,C=CCC(C(=O)NCC1(O)CCN(C(c2nc(C(F)(F)F)sc2C)=O)C1)C(C)C 30430,CC(C)(O)C(F)(F)CNC(=O)C(CNC(=O)Cn1cccc1)CC1CCCC1 30431,c1(C(CN2CCN(CCN=[N+]=[N-])CC2)=O)cc2c(F)ccc(F)c2s1 30432,c1(C(=O)OC)ccc(C(=O)NC(C)CNC(=O)C(=O)NCC2CC2)nc1C 30433,c1(OC)ccc(C(CNC(C2(CF)CC2)=O)NC(=O)CCCc2ncco2)cc1 30434,c1(C(=O)NCC2N(C(C(C)CO)=O)CCC2C)cnc2c(c1)CCCO2 30435,N1(C(CC(C)OC)=O)CCCC(C2CN(C(=O)Cc3cc(F)ccc3C)C2)C1 30436,CN1CCCCC1CC(=O)NC1CC1C(=O)Nc1ccccn1 30437,c1(C(=O)NC2CCCC(CNC(C3CC3CF)=O)C2)cn2ncccc2n1 30438,C1(NC(C2CCCOC2)=O)(CO)CCCN(C(c2cnn[nH]2)=O)C1 30439,C(=O)(CC(C(F)F)C(C)(C)C)N1C(C)CC(NC(c2cc(C3CC3)on2)=O)C1 30440,C1(C(=O)NC2(CC)CC2)CCN(C(=O)Cc2csc(Cl)n2)C1C(C)C 30441,C(=O)(C1=CS(=O)CCC1)N1CCC(NC(C2C(F)(F)C23CCC3)=O)(CF)C1 30442,C1(NC(CCOC(C)C)=O)CC(NC(c2cc(O)cc(F)c2)=O)C12CCOCC2 30443,C1(CCOC)(NC(C(C=CC)O)=O)CCN(C(c2cc(C)oc2CC)=O)CC1 30444,C1(CCNC(CSCCC)=O)C(C)CCCN1C(c1cc(=O)cc[nH]1)=O 30445,c1(C(N2CCC(C)(CNC(CN(C)C)=O)CC2)=O)ccc2c(c1)C(C)(C)CO2 30446,C1(C(N2CCC(C)(NC(CCc3n(C)cnc3)=O)C2)=O)C2Cc3ccccc3C12 30447,C1(NC(c2nc(C)oc2)=O)CCC2CN(Cc3csc(-c4ccco4)n3)CC2C1 30448,NC(Cc1ccccc1Br)CC(=O)NC(c1ccccn1)C(N)=O 30449,CC(C)C(C)(O)C(=O)N1CCC(CCC(=O)NC(CN(C)C)CCO)C1 30450,C1(C(=O)NCCCNC(c2cc(C3CC3)nc(O)c2)=O)CCc2nncn2C1 30451,c1(CN(CCC#C)CC)cc(OC)c(OC)c(Br)c1 30452,O=C(NNc1ccc(S(=O)(=O)NC2CC2)cc1)C1CCCC(c2ccccc2)O1 30453,C1(CCNC(=O)NCc2ccc(I)o2)CCN(C(c2ccccc2)=O)CC1 30454,C1(C)(C(N2CCC(OCCNC(c3c(CC)noc3C)=O)C2)=O)CCC(F)(F)C1 30455,C1(NC(c2cnc(C(F)F)s2)=O)CN(C(=O)C2=CCCC2)CCC1F 30456,C1(OC)CCOCC1NC(=O)C(c1ccc(Br)cc1)(C)N 30457,C1(CCC(C)(C)NC(C2CC2(F)F)=O)CCN(C(=O)COC(=O)CO)CC1 30458,C=Cc1ccc(CNC(C23CC2CN(C(C2Cc4ccccc4O2)=O)C3)=O)cc1 30459,C(=O)(C(F)C1CCOC1)N(C)CCOCCCN(C(=O)CNC=O)C 30460,CC1CN(C)CC1C(=O)NC1(CCNC(c2ccc(C3CCOC3)s2)=O)CCC1 30461,c1(C(=O)NCC#CCNC(COCc2onc(C)n2)=O)c2c(nn1C)CCSC2 30462,C(=O)(CCCCN=[N+]=[N-])N1CCCC(CC(N2CC(C)N(CCO)CC2)=O)C1 30463,CN1CCC(C(=O)NC2(CCCC3CC3)CC2)C1.c12ccc(s1)[nH]c2=O.C(=O)N 30464,c1(C(=O)NC(C2CN(C(C3CC3(C)C)=O)C2)C)ccc(N(C)C)cn1 30465,C1(CNC(c2cnn(C(C)C)c2N)=O)CCN(C(=O)CSC(F)F)C1(C)C 30466,N1(C(C2CC(CNC(C3N(C)CC(O)C3)=O)C2)=O)CC(O)CC12CCOC2 30467,C#CCCCC(C)Oc1c(C2(Oc3ccccc3)CCCC2)cccc1 30468,N1(C(CC(=O)NC)=O)CC2C(CNC(C3(c4ccccc4F)CC4(CC4)C3)=O)C2C1 30469,Nc1ccc(C(N2CC(CC(N3CCC3CO)=O)C3(CC3)C2)=O)nc1F 30470,C1(C(N(CC)Cc2nc[nH]n2)=O)CC(F)CN1C(=O)Cc1ccc(C(C)(C)C)cc1 30471,c1(C(=O)NCCCCCNC(C(N2CCOCC2)C)=O)cc(O)ncc1Br 30472,Cc1cc(=NCc2n[nH]c3c2CCC3)[nH]c(=NCc2ccc(C(F)(F)F)cc2)[nH]1 30473,C=CCC(C(=O)NC(C)CNC(=O)C(c1ccc(Cl)nc1)(C)C)C(C)C 30474,N1(C(Cc2c(C)nc(C)s2)=O)C(CC(=O)NCC23CCCC2CCC3)C2CCCC12 30475,c1(C(C(=O)NCC(C)N(C(=O)Cc2ccccc2F)C)=O)c[nH]c2ccccc12 30476,c1(OC)ncnc(C(N2CCC(CF)(NC(=O)CC3CC4CC4C3)C2)=O)c1F 30477,C1(C(N2CCN(C)CC2)=O)CCC2(CC2)N1C(=O)CCc1nc(Br)n[nH]1 30478,C1(NC(CC=C)=O)CN(C(=O)Cc2c(Cl)cccc2Cl)CC12COC2 30479,N1(C(c2ccn3cncc3c2)=O)CC2CCN(Cc3cnc(Br)c(F)c3)CC2C1 30480,c1(N2CCCC(CNC(c3cc(C(C)C)nn3C)=O)C2)cc(S(C)(=O)=O)ncn1 30481,C(=O)(C(C)(C)CC(F)F)NCC(C(C(C)C)C)NC(c1ccsc1Cl)=O 30482,C1(C#N)(C(=O)Nc2nn(C(C)C)c(C(=O)O)c2)CCOCC1.COC 30483,N1(C(CSCC#C)=O)CC(N(C)C)C(CNC(=O)CC(C=C)c2ccccc2)C1 30484,Cc1cncc(C(=O)NC2CCC(NC(C3CN(C4COC4)C3)=O)CC2)c1C 30485,CCC(CCO)CN=c1nc(N2CCCC(CC(C)C)C2)c2c([nH]1)CCCC2 30486,CC1(C)CCC(C(N2CC(C#N)C2)=O)CN1C(=O)CCc1ccncn1 30487,CC(C)C(C)(CN=c1cc(F)nc[nH]1)NC(C1CCN1C1CCCC1)=O 30488,c1(CN2C(C(=O)Nc3ccc(C)nc3)C=CC2)ccc2c(c1)CCCC2 30489,C12(NC(c3cnc4n3CCS4)=O)CCCCCC1N(C(C1CCOCC1)=O)CC2 30490,c1(C(=O)NCC2N(C(C(CSC)O)=O)CCCC2)[nH]c2ccc(C)cc2c1Cl 30491,N1(C(C2CCC(=O)C2)=O)CCc2ccccc2C(NC(=O)Cc2ccc(Cl)s2)C1 30492,N1(C(c2c(CNC(C(c3cnn(C)c3)C)=O)occ2)=O)CCCN(C)CC1C 30493,Cc1cc(=NCCC2CCCCN2C(c2ccc(C)c(Cl)c2)=O)[nH]c(CO)n1 30494,C1(OC)CCCC(CC(N2CCCCC2C(C)NC(=O)C(C)C)=O)C1 30495,c1(-c2nc(C(CC)C)nn2C23CC(C2)C3)ccc(Cl)c(S(C)(=O)=O)c1 30496,c1(CO)cc2cc(-c3nc(-c4ccc(SC(F)(F)F)cc4)no3)ccc2[nH]1 30497,N1(C(C=CS(C)=O)=O)CCN(C(c2ccccc2C(N)=O)=O)CC1c1cn[nH]c1 30498,c1(CCC)cccc(OC(C2CC2c2cccs2)=O)c1 30499,Cc1nn(C2CC2)c(C)c1C(N1CCCC(NC(=O)CC(F)(F)F)C1)=O 30500,N1(C(CC(C)SC)=O)CC(NC(c2cc(C)cc(F)c2)=O)CC(F)C1 30501,c1(C(N(C(C)CNC(=O)C(F)(F)C(F)F)CC)=O)ccc2c(c1)COC2 30502,N1(C(c2cc(C)nn2C)=O)CC(CO)C2(C1)CN(c1nc(C)nc(C)c1F)C2 30503,C(=O)(CC(C)CC(C)(C)C)NCCC(=C)CNC(=O)CS(=O)(=O)N1CCCCC1 30504,c1(CCN(C(=O)C(C2CCN(C(=O)OC(C)(C)C)C2)F)C)cc(F)cc(F)c1 30505,c1(N2CCC(C(C)C)CC2)[nH]c(=NCC23CC2CN(C)S3(=O)=O)nc2sccc12 30506,C1(C(=O)NC2(C)CC(NC(c3c(C)ocn3)=O)C2)CCOC2(CCC2)C1 30507,N1(C(Cc2ccc(C)cc2)=O)CCCC(C(=O)NOCC(O)C(C)C)C1C 30508,c1(C(=O)NCC2(NC(CC(CCC)(C)C)=O)CCCC2)c(F)ccc2nc[nH]c12 30509,C(=O)(C(F)C(C)C)NC(CCOC)CNC(c1ccc(CN2CCCCC2)s1)=O 30510,c1(C(N2CCC(CC)(NC(c3cnoc3)=O)CC2)=O)ccc2c(c1)nc(O)n2C 30511,C1(CC(=O)N(CC(CN(C)Cc2sccc2Br)O)C)CC(C)(C)CO1 30512,CCC(C)(CNC(C1(C(C)C)CCN(C(=O)CC(C)SC)C1)=O)CO 30513,C1(NC(C2SC3C=CC2C3)=O)CC2CCC1N2C(=O)C1=C(Cl)CCC1 30514,CC(O)(C(=O)NCC(CNC(C1CN(CC(F)(F)F)C1)=O)CO)C1CCC1 30515,C(=O)(CC(C)C(F)(F)F)NCC1=CCCN(C(C2=CCCC2C)=O)C1 30516,C1(CC=C)(C(=O)N(CC(=C)C)C)CN(C(C2C=C(C)CS2)=O)C1 30517,C(C(CC(F)(F)F)NC(=O)CC(CC1CCCC1)CC)NC(COCCC)=O 30518,C1(C(C)(C)CNC(C2COC(=O)N2)=O)CCN(C(C2CCC23CCC3)=O)CC1 30519,CC(C)(CC(=O)NC1CN(C(=O)CC2CCn3cncc3C2)CC1F)C(F)F 30520,C(=O)(C1CCCc2nccn21)NCCN(C)C(c1nc2ncccn2n1)=O 30521,C1(NC(CC(=O)NC)=O)CCC(N(C(=O)C=CC(N)=O)C)CC1 30522,S(=O)(=O)(c1cc(C)c(Cl)cc1F)N1CCCC(CCNC(C=C(C)C(=O)O)=O)C1 30523,Cc1cc(=NCC2(NC(=O)CC3(CO)CC3)COC2)[nH]c(-c2cccnc2)n1 30524,C(=O)(CCCCCC#N)NCC(CC)(CC)c1ccc(Cl)cc1 30525,c1(C(N2CC3C(CNC(=O)C=CC4CC4)C3C2)=O)ccc(F)c(F)c1 30526,Cn1ncc(C(=O)NCCNC(C2COC(C)(C)C2)=O)c1C#N 30527,CC1CC(C(N2CCCC(CN=[N+]=[N-])C2)=O)CN(C(=O)CCNC(=O)CO)C1 30528,c1(N(CCN2CCC(CC=C)(NC(=O)CC(C)CC)C2)C)c(Cl)cc(Cl)cc1Cl 30529,C1(C(N2CCN(Cc3ccc(Br)s3)CC2)=O)CC2CC2N1C(C1CCCO1)=O 30530,N1(C(c2ccnc(C)n2)=O)CC2C3CCC(C2C1)N(C(C1(N(C)C)CCC1)=O)C3 30531,CC1CCC=C1C(=O)NCCC(O)CNC(=O)CC1CCCCCCC1 30532,C1(C(=O)NCCC2(OC)CN(C(c3ccccc3C(N)=O)=O)C2)CC(O)C(F)C1 30533,c1(OC)ccc(Cl)c(C(=O)NCCC2(NC(C3CCC(C4CC4)C3)=O)CC2)n1 30534,C(CS(=O)(=O)CC(=O)NC1CCC1CNC(=O)Cc1scnc1C)OC 30535,N1(C(c2ccc(CC)s2)=O)CCC(CC(C)NC(=O)CN2C(C)CCC2C)CC1 30536,c1(OC)ccc(C(N2CC(N(C(=O)CC3CCOC3(C)C)C)C2)=O)c(C)c1 30537,C1(CNC(C(C)NC(CC)=O)=O)(CNC(=O)CSC(F)(F)F)CC12CCC2 30538,c1(C(N2CCN(C(CCOCC)=O)C(CCO)C2)=O)oc2ccccc2c1CC 30539,C(=O)(C(C)(C)CS(N)(=O)=O)NCC1CN(C(c2c(CC)ncs2)=O)C(C)C1 30540,c1(-c2scc(C(=O)Nc3cc(C)[nH]n3)n2)cncc(N2CCCC2)c1 30541,c1(CN2CCCC(CC(=O)Nc3c(C(N)=O)nccn3)C2)ccc2c(c1)CCO2 30542,c1(C(=O)NCC2(C(C)NC(C3=CCCC3C)=O)CC2)ccc(F)cc1[N+](=O)[O-] 30543,C1(CN(C(CCN(C(c2nccn2CC)=O)CC)=O)C)CCOC1C 30544,c1(C(N2CC(O)CC(NC(CC=CC=C)=O)C2)=O)nc2ccccc2nc1C 30545,CC(C)(C(=O)NCCCCNC(C1(C(C)(F)F)CC1)=O)c1cncs1 30546,C(C(C(=O)NCc1ncc(CO)o1)NC(=O)C=CC1CC1)N(C)C 30547,N1(CC(C)(C)NC(C(CC)OC2CCCCC2)=O)CCN(C(C2CC2C)=O)CC1 30548,C1(C)(C(=O)NC2C(N(C(CCOCCC)=O)C)CCCC2)CCCCCCC1 30549,C(C1CCCCCC1)=CC(=O)NCCCC(C)NC(C1CC(C(C)C)C1)=O 30550,N1(C(c2c(CC)[nH]nc2Cl)=O)CCC(NC(=O)CCc2cccc(C)c2)C(C)C1 30551,C(C)(CCCC(=O)NCC1CCC(O)C1)NC(C(C)C)=O 30552,c1(CC(=O)NCC(CC)NC(=O)CSCCN(C)C)scnc1C 30553,C(=O)(CC(C)CC(=O)NC1CCN(C(C2(C3CC3)CCOCC2)=O)C1)OC 30554,C(C(N=c1[nH]nc(C#N)s1)C(C)C(C)C)NC(c1c(F)cc(OC)cc1F)=O 30555,C12(C(=O)NCc3c(CN)cc[nH]3)CCC1CN(Cc1ccccc1)C2 30556,N1(C(C=COCC)=O)CCOC2CCN(C(=O)C=CC(C)C)CC12 30557,N1(C(c2cc(C)on2)=O)CCCC(C)C1CCN(C(=O)CN1CCCS1(=O)=O)CO 30558,C(=O)(C(C)CC(F)F)NC(C(=O)NCCc1cnc(C)[nH]1)CO 30559,CC1CCN(CC2CCCC(=O)N2)CC1NC(c1ccsc1-n1cnnn1)=O 30560,C12(C(=O)NC(CNC(c3nc(OCC)oc3)=O)(C)C3CC3)CCCCC1C2 30561,CC1CCC(C(=O)Nc2cncnc2)CN1C(=O)C(=O)N(CCC(N)=O)c1nccs1 30562,c1(NC(C2(NC(CN(C)C(=O)C3CC3)=O)CC2(C)C)=O)ccc2ccoc2c1 30563,C(C(C(=O)NC1COCC1NC(=O)C(C)(C)c1cccnc1)N(C)C)OC 30564,N1(C(Cc2cn(CC)nn2)=O)CC(F)CC1C(=O)NCc1csc(C)c1 30565,N12CCC(F)(F)C(C1)C2.c1(OC)cc(COC(c2sc(Br)nc2C)=O)ccn1 30566,CC1CCN(C(=O)CC2N(C(=O)CN3CCSCC3)CCC2(C)C)CC12CCC2 30567,CC1(C)CCN1CC(=O)NC1CCCC1NC(C1(c2cccnc2)CCCC1)=O 30568,C(CC(C(C)C)NC(=O)CCNC(N)=O)NC(C1CC(C(F)F)(OC)C1)=O 30569,c1(C(C)C)ccc(CCC(=O)NC(C)C(CO)NC(=O)COC2CCC2)cc1 30570,c1(CC(N2C3C(NC(c4coc(CO)c4)=O)CC(C3)C2)=O)cn2c(n1)CCCC2 30571,C1(C(=O)NCC2(C(=O)OC)CCC2)C=CC(NC(=O)CC2CC(=O)C2)C1 30572,Cc1cnn2cc(C(N3CC(O)CC3c3ccc(F)cc3)=O)cnc12 30573,CC1CN(C(=O)CCSC2CCCC2)CCCN1C(C1CSCCS1)=O 30574,C1(C(=O)NC2CC(CC(=O)NC3CC(F)(F)C3)C2)CCCCC1F 30575,C1(CNC(c2c(OC)nn(C)c2)=O)CN(C(c2cc(OC)no2)=O)CC(C)(C)O1 30576,N1(C(CSCC(C)=O)=O)CC2(CCC2)CC1CNC(c1nn[nH]c1C(F)(F)F)=O 30577,c1(C(=O)NC(CN(C(=O)CC(C)n2ccnc2)CC)C)ccc(Cl)c(C)c1 30578,O(C1CCCc2ccccc21)CC(=O)NC1CCN(C(c2cnc(C)o2)=O)C1C 30579,C1(CCCNC(CNS(NC)(=O)=O)=O)CN(C(=O)CC2CSC2)CCO1 30580,C1(NC(C2(CCNC(C3C=CC=CC=C3)=O)CCC2)=O)CC2CCC(C1)S2 30581,N1(C(c2ccc(CNC(C(CC)COC)=O)cn2)=O)CC(O)CC1(C)C 30582,c1(C(=O)NCC(N(C(CC(CCC)C)=O)C)C2CC2)cnc2scc(C)n2c1=O 30583,N1(C(CC)=O)CC(NC(c2ccc(S(=O)(=O)NCCO)s2)=O)CC(C)(C)C1 30584,C(C(C(=O)NCCc1cn[nH]c1)C(C)C)NC(C1CC(CCC)C1)=O 30585,C(N=c1cc(CC(C)C)nc[nH]1)C1CN(C(C(C=C)c2ccccc2)=O)CC1C 30586,c1(C(=O)NC(C2N(C(C(C)c3cncs3)=O)CCC2)C)n[nH]c2ccc(Cl)cc12 30587,Cc1cnnc(O)c1C(=O)NCCCCC(C)NC(=O)CC(C)NC(N)=O 30588,c1(C(N(CCCCNC(c2cn(C)cn2)=O)C)=O)cc(OC(F)F)n(C)n1 30589,C(=O)(C1=NOC2(CCC2)C1)N1CCC(NC(=O)C2=CCC(C(F)(F)F)OC2)C1 30590,N1(C(CSC)=O)CCN(C(=O)C(CC(C)C)OC(C)=O)CC12CCC2 30591,CC1(C)CCC(C(=O)NCC2(C)CCCN(C(c3ocnc3C(F)F)=O)C2)OC1 30592,c1(CNC(CC2CCC(NC(C3CN(C(C)=O)C3)=O)C2)=O)ncccc1Cl 30593,c1(OCCCC(=O)NCC2CCN(C(C(CSC)C)=O)C2)cccc([N+](=O)[O-])c1 30594,Cc1cc(C(N2CCCC(CC(=O)NC3CN(C)CC3C)CC2)=O)cnc1O 30595,N1(C(c2c(C)nsc2)=O)CC2COCC2(CN2CCC(C3CC4C=CC3C4)C2)C1 30596,C12=NC=CC(=NCc3ccc(F)cc3CN1)N2.O=S(=O)(CC1CC1)C1CC1 30597,C12(C(N3CC(NC(C4(OC)CCOCC4)=O)C3)=O)CCOC1CS(=O)(=O)C2 30598,c1(C(=O)NCC2C(NC(c3cncc(NC)c3)=O)C2)c(F)ccc(F)c1Cl 30599,c1(OC)ccc(CC(=O)Nc2cccc(C(=O)O)c2F)c(F)c1F 30600,C(=O)(C(F)C(C)CNC(c1ccsn1)=O)N(C(C)C)CCN(C)C 30601,c1(C(N(C2CC(C(=O)NC3CC3(F)F)C2)C)=O)ccccc1S(C)(=O)=O 30602,C=CCC(C(=O)NC(C)CCN(C)C(c1cnn(C)c1OC)=O)C(C)C 30603,c1(OC)ccc(C(N2CCC(CNC(c3c[nH]nc3OC)=O)C(C)C2)=O)c(O)c1 30604,C1(NC(COCCSC)=O)CC12CCN(C(c1csc3cncn13)=O)CC2 30605,c1(CC(=O)NC(CCNC(CC2(C(=O)OC)CC2)=O)C)c(C)n[nH]c1C 30606,C1(C(=O)NC(C2(O)CCCCC2)C)CCC(C)(C)N(C(=O)CN2CCCC2)C1 30607,c1(C(=O)NCC2(C)N(C(=O)C=CC(C)C)CC(OC)C2)cc2cnn(C)c2s1 30608,N1(C(C2CCN(C(CC)=O)CC2)=O)CCC(CNC(C2CC(OC)C2)=O)C(O)C1 30609,N1(C(C(C)NC(=O)NC)=O)CCCC(C(=O)NC2CCC(O)C2)C1 30610,C(CCCCCNC(c1cccc(C2CCOC2)c1)=O)NC(=O)C(=O)NC1CC1 30611,Cc1[nH]nc(C(=O)N(C)CCOCCCN(C(=O)Cc2ccnn2C)C)c1Cl 30612,N1(C(c2c(C)c(Br)cnc2)=O)CCCN(C(=O)C(C)NC=O)CC1C 30613,Cc1noc(C)c1C(=O)NCC(=O)NC(C1CCCCC1)(C)C 30614,n1(C(C(=O)N(CCNC(c2c(C)ccnn2)=O)C(C)C)C)cnc2ccccc12 30615,CC1=C(C(=O)N2C3CCC(C3)C2CC(N2CCCCC2C(F)F)=O)CCC1 30616,c1(C(N(C2CCN(C(C3CCCOC3C)=O)C2)CC#C)=O)cc(C(N)=O)nn1C 30617,c1(CCC(=O)NC(C2CCCC2)CNC(COCC=C)=O)cnn(C)c1 30618,n1(CC(=O)NCCCCC2CN(C(C=CCC)=O)C2)cnnc1C(C)C 30619,C1(NC(Cc2cnc(C)s2)=O)CC2CC1CN(C(C1(O)CC1)=O)C2 30620,C1(CNC(C2(CSC)CC2)=O)CCN(C(=O)Cc2cccc(C)c2)C12CCC2 30621,C1(NC(C2CN(C)C(=O)C2)=O)CC12CCN(C(c1conc1C(C)(C)C)=O)CC2 30622,CCC(=O)CCC(=O)N(CCCCN(C)C(c1cocc1C(N)=O)=O)C 30623,N1(C(C(C)SCCCC)=O)CC(C2CC2)(C(=O)NCc2csc(C)c2C)C1 30624,C1(NC(C=NOC)=O)CCC2(CCN(C(=O)CCc3ncc(F)cn3)C2)C1 30625,c1(C(=O)NCC(C(=O)OC)C)cncc(CNC(=O)C(c2cnn(C)c2)O)c1 30626,N1(C(C2N(CCC)CCC2)=O)CCc2ccccc2C1CNC(c1ccns1)=O 30627,c1(CC#N)ccc(NC(C2CCN(Cc3cccc(Br)n3)C2)=O)cc1 30628,C1(NC(C2CCN(C)C2)=O)CCC12CN(C(=O)C=CCF)C2 30629,N1(C(C(CCC)NC(C)=O)=O)CC2CCC(NC(=O)CSC(F)(F)F)C2C1 30630,Cc1snnc1C(=O)NCC(C)N(C(=O)CC1(Oc2ccccc2)CC1)C 30631,N1(C(C(CCC)CNC(c2nccnc2N)=O)=O)Cc2nncn2C(C)C1 30632,N1(C(CCC(=O)NC)=O)CC(NC(C2(C(F)F)CCCCC2)=O)CCC1C 30633,Cc1cccc(C(=O)NCC2(O)CCCN(C(=O)C(CO)C(C)(C)C)C2)c1C#N 30634,CCC(F)(F)C(=O)N1CCC(C(C)CNC(=O)CCC2CC(F)(F)C2)CC1 30635,N1(c2nc(NC(c3ncc[nH]3)C)c3c(n2)scc3)CCOC2(CCSC2)CC1 30636,N1(C(CC2CCN(C(c3cc(C)c(O)nn3)=O)C2)=O)CC2CCC1C(C(=O)O)C2 30637,S(=O)(=O)(c1ccc(C(=O)O)nc1)NC(C(c1ccccc1)OCC)=O 30638,N1(C(c2c(OC)csc2)=O)CC(CNC(C2CC(=C3CCC3)C2)=O)C(O)C1 30639,c1(C(=O)NCCN(C(c2c(CCC)nns2)=O)C(C)C)cccc2ccncc12 30640,c1(C(N2C(C(C)NC(CNC(CC)=O)=O)CCCC2)=O)cc(C)n(C(C)C)c1C 30641,C(=O)(C#CC1CCOCC1)N1CC(CCCCNC(c2n(CC)c(O)nc2)=O)C1 30642,C(=O)(CCC(=O)C(C)(C)C)N1CCC(C)C1CNC(=O)C(c1ccccn1)C 30643,N1(C(c2c(COC)noc2)=O)CC2CCN(C(c3cc(N)ccc3C)=O)C2C1 30644,CC(C)C(C)C(CNC(=O)COC(F)F)NC(c1cc(N)ccc1F)=O 30645,C(=O)(C(C)(F)C(F)(F)F)NC(C1CCN(C(C2(C(=O)NC)CC2)=O)CC1)C 30646,S(=O)(=O)(c1cccc(C(=O)NC23CC(NC(=O)Cc4conc4C)(C2)C3)c1)NC 30647,Cc1cc(C(=O)N(CC(=O)NCC2CC(C)CO2)C(C)C)nn1C 30648,c1(CC(=O)NCC(CC)NC(C(CCC)NC(N)=O)=O)cc(Cl)cc2c1OCC2 30649,C(CNC(c1ccc(C(N)=O)cc1)=O)(C(C)(C)C)NC(c1cnc(COC)s1)=O 30650,N1(C(C(C(C)(C)C)O)=O)CC2(C(=O)NCCn3ccnc3)CCC1CC2 30651,C1(NC(C2(COC)CC=CC2)=O)C2CCN(C(C3CC(C)(C(=O)O)C3)=O)CC12 30652,c1(CC(=O)NC(C2CCCO2)COC)cccc(NCc2ccccc2Cl)c1 30653,C1(NC(c2n[nH]c(C)c2C)=O)CC2CC(NC(=O)CCn3cccc3)CC2C1 30654,Cc1nc(C(C)C)ccc1C(=O)N(C)CC1(O)CN(C(=O)COc2ccon2)C1 30655,c1(C(=O)NCC(C)N(C)C(c2cnco2)=O)c(F)ccc(N)c1Br 30656,CCC(F)(F)CC(=O)NC1CN(C(c2n[nH]cc2C(F)(F)F)=O)CC1(C)C 30657,N1(CCCNC(c2cscn2)=O)CCN(C(c2cnn[nH]2)=O)CC1 30658,c1(CNC(C2(COC)CC2)=O)cc(C)c(C(=O)NCCN2C(=O)CCC2=O)o1 30659,N1(C(CCOCC(C)C)=O)CCC(C(C)NC(=O)C(F)(F)c2ccncc2)CC1 30660,C1(F)(CNC(C=C(C)C(C)C)=O)COCCN(C(=O)CC2(CS(C)(=O)=O)CC2)C1 30661,S(=O)(=O)(c1cccnc1)NCCC(=O)NCC1C(CNC(=O)C2=CCC2)C1 30662,Cc1cncc(NC(=O)Cc2ccc(O)nc2)c1 30663,C(=O)(CCCCN(C(=O)C(C)(C)C1(O)CCC1)C)NCC(C)CCO 30664,S(=O)(=O)(c1ccc(=NCCCC(F)(F)F)[nH]c1)N(C1CC(C)OCC1)C 30665,c1(C(N(C2CCCN(C(C3CCCC34CC4)=O)C2)CC)=O)ccc(C)cc1C 30666,CC(C)C(C(=O)N1CCN(C(c2ccc(F)cc2)=O)CC1)NC=O 30667,C(=O)(CC(O)C1CCCC1)NCCN(C)C(=O)NCC1(C(=O)N)CC1.C(C)(C)C 30668,c1(OC)ncccc1C(=O)NC1CN(C(c2cncc(C(C)(C)C)n2)=O)CC1O 30669,N1(CC(=O)N(C2CC(C)(C#N)C2)C(=O)C2CC2)CCC2CCC12C 30670,c1(C(=O)NCC2C(NC(c3cnc(OCC)nc3)=O)C2)c(F)ccc2nc[nH]c12 30671,C(=O)(C(CCC(N)=O)n1cc(-c2cncc(Cl)c2)nn1)N(C(C)C(F)F)C 30672,N1(C(c2nc(CS(C)(=O)=O)oc2)=O)CCN(C(c2cncc(O)c2)=O)C2(CC2)C1 30673,c1(C(C)=O)ccc(C=CC(=O)NCC(C)(C2CC2)NC(=O)C(C)CF)cc1 30674,Cc1c(C(=O)NC2C=CCCC2C(=O)NCCCNC(N)=O)nnn1C 30675,c1(C(=O)NCC2CCN(C(C(C)(CO)OC)=O)C2)cc(Cl)c(F)cc1N 30676,CCCCC(=O)C(=O)NCC1CN(C(C2CC23CCOCC3)=O)CCO1 30677,c1(CC(=O)N(C(c2ccccc2)CNC(=O)Cn2nccn2)C)nnc(O)s1 30678,c1(-c2ccc(CC)cc2)ccc2[nH]cc(C(N3CCCC(C(=O)OC)C3)=O)c2c1 30679,C1(NC(C(=O)N(CC(N)=O)C)=O)CCN(c2ncccn2)C1 30680,C=CC1(C(=O)NC(C)CCc2cn[nH]c2)CCN(C(c2ccn(C)c2)=O)C1 30681,c1(C(=O)NCC2(NC(CC(CC)C3CCC3)=O)CCOCC2)ccc(N)cc1Cl 30682,N1(C(C2CC(C(C)C)C2)=O)CC(NC(c2ccccc2C(N)=O)=O)C(F)C1 30683,O(NC(=O)C(CCF)NC(=O)CC12CCCC1C2)C(CC)CC 30684,c1(C(=O)NCC2(CN3CCN(C(=O)C4CC4)CC3)CC2)ccc2nncn2c1 30685,Cc1nc(C)n(CC(=O)NCC2CCN2C(=O)C(F)CC2CCOC2)n1 30686,N1(C(c2c(OC)nccn2)=O)CCCN(Cc2ccc(Cl)cc2O)CC1C 30687,c1(C(N2CCC(C)(NC(C34CCC(OC)C3CC4)=O)C2)=O)cc(F)c(F)cc1F 30688,c1(C(N2CC(N(C)C(c3cc(C4CC4)ns3)=O)C2)=O)ccc(-n2cccn2)nc1 30689,C(=O)(CC(O)CC(C)(C)C)N1C2C(N(C(CCCCCCC)=O)C)CC(C2)C1 30690,C1(C(=O)NCC(C)N(C(=O)C(=O)NCC2CC2)C)CC2CSCC(C1)C2 30691,C1(CCNC(=O)C(c2ccc(F)cc2)O)CSCCN1C(C1CCS(=O)CC1)=O 30692,C(C(C)(CO)NC(=O)CCCNCCn1cnccc1=O)NC(C1C(C)(C)C1)=O 30693,C1(C(N(CCC(C(C)C)NC(=O)C(C)c2ccco2)C)=O)CN2CCCN1CC2 30694,Cc1cc(C(=O)OC(C)(C)C)n(-c2ccccc2)n1.C12CCOC(C1)CNC2=O 30695,C#Cc1ccc(C(=O)N(CC(O)COC)C)c(C)c1.c12ccc(s1)C(=O)NC2 30696,Cc1c(C(=O)NCC(C2CC2)NC(=O)Cn2nccc2C)cnn1C1CCCC1 30697,C12(CNC(=O)CC3CC3(Cl)Cl)CC3CC(CC(NC(=O)C(O)C(F)(F)F)(C3)C1)C2 30698,N1(C(C(C(CC)O)C)=O)CCN(C(c2cc(C)c(C(F)F)cn2)=O)C2(CC2)C1 30699,CC1CN(C(C2CCC3(CCC3)C2)=O)CCCN1C(=O)CCc1cn(C)nn1 30700,C12(C(N(CCN=[N+]=[N-])CC)=O)CC1CCN2C(=O)CC1CC2CC2C1 30701,n1(CCS(CC)(=O)=O)c(=NCCc2sc(N(C)C)nc2C)[nH]c2cc(Cl)ccc12 30702,C1(C(C)CO)CCN(C(=O)C(c2ccnn2C)NC(=O)CCN(C)C)CC1 30703,N1(CCC(N2CCC(C)(C)C(CO)C2)=O)C(=O)C2CC=CCC2C1=O 30704,COn1cnc(C)c1C(=O)NC1CC1CNC(c1cc(C)ccc1C1CC1)=O 30705,C1(CCNC(c2ccc(Cl)s2)=O)CCN(C(=O)COc2cccc(O)c2)CC1 30706,C(C(=O)NCCC(=O)NC)(NC(COCCC)=O)C1CC1 30707,c1(C(=O)NC2C(NC(c3nnc(C)s3)=O)CCC2)cccc2c1COC2 30708,c1(C(=O)NCCN(C(=O)C(F)CC2CCC2)CC)ncncc1Cl 30709,CC1Cc2ccccc2N1CC1CC2CCCC2N1 30710,N1(C(C(CC)NC(N)=O)=O)CCN(C(c2n[nH]c(O)n2)=O)CC1c1cnn(C)c1 30711,n1(CC)cc(CN2CCC(CC(N3CCCC(CN(C)C)C3)=O)C2)c(C)n1 30712,c1(C(C2CCOC2)OCC)nc(-c2ccccc2)nn1-c1cnn(C)c1 30713,c1(OC)ccc2nc(C)c(C(=O)NCC3CCC3NC(=O)Cc3ccsn3)n2n1 30714,C1(NC(c2c(CC)nns2)=O)CN(C(=O)CSc2cccc(C)c2)CCC1C 30715,C1(C(N2CCC(CCNC(C(C=C)(F)F)=O)CC2)=O)CN2CCC1CC2 30716,Cc1cnc(C(=O)NC2CCN(C(=O)C(=CC3CCCCC3)F)C2(C)C)cc1C 30717,Cc1ncc(C(=O)NC2(C)CCCN(C(c3c[nH]c(Br)c3)=O)C2)c(=N)[nH]1 30718,c1(C(N2C(CNC(C(C)Oc3cccnc3)=O)CCCC2)=O)cccc(N)c1O 30719,N1(C(Cc2nc(C)[nH]n2)=O)CCCC12CCN(C(=O)CCc1nncn1C)CC2 30720,C(=O)(CC(O)(C(F)(F)F)c1ccc(C)o1)NC(CNC(C=C(CC)CC)=O)C 30721,C1(C)(C2CCCN(C(C(=O)NC(C(=O)OC)C)C3COC3)C2)NC(=O)NC1=O 30722,C1(NC(=NCCSC)NCCc2cccc(O)c2)CCOC2(CCSC2)C1 30723,N1(C(c2cc(CC)[nH]n2)=O)CCC=C(C(=O)N2CC3CCC2CO3)C1 30724,n1(CCC)ncc(CN2CC(CC(=O)NC3CSC3)C2)c1C 30725,c1(C(N2CCCCC(NC(C(CCC)C#N)=O)C2)=O)noc2ncccc12 30726,c1(C(N2CC=CC(NC(=O)Cn3ccc(C4CC4)n3)C2)=O)cc2c[nH]cnc-2n1 30727,C(=O)(CC(O)CC(C)(C)C)N1CC(SC)C(NC(c2ccncc2)=O)C1 30728,C1(C(=O)O)C=CCN(Cc2ccc(N3CCCC3)nn2)C1 30729,c1(C(C(=O)N2CC(N(C(Cc3cnc(C)[nH]3)=O)C)C2)(F)F)cccc(F)c1F 30730,C1(C(=O)NCc2ccc(C#N)o2)(NC(CC=CCCCCC)=O)CCCCC1 30731,c1(C(N2CCCC2)=O)ccc(Cl)c(S(=O)(=O)N2C3CCCC2CC(O)C3)c1 30732,C1(C(N)=O)C2CC3CC(C2)CC1(NC(NC1CCCc2c[nH]nc21)=O)C3 30733,C1(OC)(CNC(C2(C)CCCCCC2)=O)CCN(C(c2[nH]c(O)nc2C)=O)CC1 30734,CC1(C#CC(=O)N2CCC3C(C2)CN3C(C2CCC(C(N)=O)C2)=O)COC1 30735,C1(NC(CCCCONC(C2C(OC)CCC2)=O)=O)CCCC2CC12 30736,C1(NC(c2ccnc(Cl)c2O)=O)CCCCN(C(=O)Cc2c(O)ncnc2O)C1 30737,C1(C(=O)NCC2C=CC(NC(C3(OC)CC3)=O)C2)CS(=O)(=O)CC(=O)N1 30738,C(C)(CC(=O)N1C(CNC(C2CCCCC2)=O)CC2CC12)(C(F)(F)F)N(C)C 30739,c1(COC)cccc(CNC(C2COCCN2C)=O)c1 30740,c1(C(=O)NC(CNC(c2nccc(C#C)c2)=O)C(C)C)ccc(F)c(C#N)c1 30741,c1(CC(=O)NCC2Cc3cc(Br)ccc3O2)ccc2c(n1)OCCO2 30742,C#Cc1cn(C)nc1C(=O)NC1CCCC(C(=O)NC(c2ccns2)C)C1 30743,C1(C(F)(F)F)(OC)CCCN(C(=NCc2ccc(C#N)cc2)NC(C)C)C1 30744,C(=O)(CCCS(C)(=O)=O)N1CCCN(C(c2c(C)ncn2C)=O)CC1 30745,CCC(O)(C(=O)NCC1CC2CC2N1C(=O)C(C)=C1CCCC1)c1ccccc1 30746,C1(NC(c2cc(C)no2)=O)CCC2CN(C(c3cncc(C(N)=O)c3)=O)CC2C1 30747,CC1CCCCN1CC(N1CCC(CCC(=O)NCCC(O)C2CCC2)CC1)=O 30748,c1(CNc2nc(-c3cn(CC=C)nc3)sc2)sc(C)nc1C 30749,C1(SCC)CCC(NC(c2c[nH]nc2-c2ccccc2Cl)=O)CC1 30750,c1(C(C)NCC(c2ccc(OC)cc2)(C)O)nc(O)c2c(C)c(C)sc2n1 30751,N1(C(C2C(OCC)C2)=O)CCC(CCC(=O)NC(C)CC2(O)CCC2)C1 30752,c1(C(=O)NC(CC)CNC(C23CC=CCN2CCC3)=O)cc(C)c2[nH]cnc2c1 30753,c1(C(=O)NC(C(C)C)C(C)NC(c2ccsn2)=O)cnc(C2CC2)[nH]c1=N 30754,c1(C(C)=O)ccc(NC(c2ccc(NC(c3cccc(I)n3)=O)nc2)=O)cc1 30755,N1(C(CCc2ccc(C)cc2)=O)CC2CC(NC(C3CCN(C)CC3)=O)CC1C2 30756,Cc1cc(C)c(CN2CCN(C(C)C(=O)NC3CCCC3)CC2(C)C)cc1C 30757,C12(NC(c3cc(OC)n[nH]3)=O)CC(CNC(=O)C(C)O)(C1)OC2(C)C 30758,C1(C(=O)NC2CCN(CC)C2)CCC(CNC(C2C3COCC23)=O)CC1 30759,C1(OC)(OC)CC(C)(C(=O)NCC(F)CNC(=O)CC2C(C)(C)C2(C)C)C1 30760,c1(C(=O)NC2(C3N(C(c4nncc(OC)c4)=O)CCC3)CC2)c(Cl)cccc1Cl 30761,c1(-n2cc(NCC3CC34CN(OC)C4)nn2)cc(C(=O)OC)ccc1C 30762,c1(CCCC(=O)N(C2CCN(C(CC=C(C)C)=O)C2)C)ccccc1Cl 30763,CCC(CC(C)C)C(=O)N1CCC(CO)C(NC(=O)CC2CCCC(C)C2)C1 30764,c1(C(N2CC3C(NC(C(CCN(C)C)O)=O)(C3)C2)=O)c(Cl)cncc1Cl 30765,Cc1cc(NC(c2cc(CNC(C3CCC(N(C)C)C3)=O)no2)=O)c(=O)n(C)c1 30766,N1(C(C(CCCC)O)=O)CC(CNC(=O)C(=C2CCCCC2)F)OC2(CCC2)C1 30767,N1(C(Cc2cc(C)on2)=O)CCC(O)(CN(C(=O)C(N2CCCC(C)C2)=O)C)C1 30768,c1(NC2CCN(CC=C)CC2)ncc(S(=O)(=O)N2CCCC(C)C2)cc1Cl 30769,CCC(CCOC)C(=O)NCC1CCC1NC(c1nccc(OC)c1O)=O 30770,C1(C(=O)NC(CC)CCO)C2CC2CN1C(=O)C(c1cccn1C)=O 30771,C(CC#CC(C)(C)C)NC(CC(CC)NC(C1(CC)CC1)=O)=O 30772,Cc1cc(C(=O)NC2CCN(C(=O)COCCCF)CC2F)cc2nc[nH]c12 30773,c1(CNC(C2COCC2NC(C2CCCCS2)=O)=O)cccnc1Cl 30774,Cc1cc(Cl)cc(C)c1C=CC(=O)NOCCOCCO 30775,c1(NCC(C)S(N)(=O)=O)ncccc1S(=O)(=O)NC(CC(N)=O)C1CC1 30776,c1(S)nncn1Cc1ccc(Br)s1.O=C1CCCN1C1CCCN1C1CC1 30777,Cc1ccc(C(N2CC3(CCN(C(c4nc(Br)c[nH]4)=O)C3)C2)=O)cc1C#N 30778,CN1CCCC(CNC(C2CSCCN2C(c2ccc(C#N)cn2)=O)=O)C1=O 30779,C1(C)(CNC(COC(CC)(C)C)=O)CCN(C(=O)CSCCN(C)C)CC1 30780,C1(C(N2CCC(N3CCN(C(=O)Cc4cnco4)CC3)C2)=O)CCCCC1(F)F 30781,C(=O)(C(C)CC(F)F)NC1CC(C(C)NC(c2ccn(CCC)n2)=O)C1 30782,CCC(C)C(=O)N(C(CNC(C1CC2CC2C1)=O)C1CC1)C 30783,c1(-c2cccc(C3C(C(=O)NC(CC(C)=O)C)C3)c2)ccc(S(=O)(=O)NC)cc1 30784,C1(NC(c2n(CC)ccn2)=O)CCCN(Cc2nnc(C3CC3)s2)C1 30785,C(=O)(N=c1nc[nH]n2cccc12)C1N(C(c2cccc(NC(C)=O)c2)=O)CCC1 30786,C(=O)(C(C)=NOCC#N)NCC1C(C(=O)NCC(COCC)C)C1(C)C 30787,CCC1=C(C(=O)NCC2CCN2C(C2CCc3n[nH]c(C)c3C2)=O)CCCO1 30788,C1(NC(c2c(C)cccn2)=O)C2COCC1CC(NC(=O)C1=NOC(C)C1)C2 30789,N1(C(C(C)OC(C)(C)C)=O)CC(C2CN(C(=O)CSC3CCCCO3)C2)C1 30790,C1(COC)(NC(=O)C(F)CC2CCCC2)CN(C(=O)Cn2cc(Cl)cn2)C1 30791,CCC(CCC(=O)NCC1(C)CC(NC(=O)CSc2ccc(C)cc2C)C1)OC 30792,Cc1c(O)c(=O)ccn1CC(N1CCCN(C(=O)C(F)n2ccnc2)CC1C)=O 30793,C1(C)(C(=O)NC2CC(CNC(C(C)OC3CCCC3)=O)C2)CCC(F)(F)CC1 30794,c1(CC(=O)NC(CCCCNC(C2(C)ON=C(C)C2)=O)C)c(C)nc(O)nc1C 30795,c1(OC)cc(CN2CC3(CC(C(=O)Nc4cccc(C)c4Cl)C3)C2)cc(F)c1 30796,C(CCCCCC(=O)NCC(O)C1(Cl)CC1)NC(C(CN(C)C)(F)F)=O 30797,C(N)(CCC(=O)N1CCOCC1)n1cc(C2(C)CC2(Cl)Cl)nn1 30798,CCCC(C(=O)N1CCCCC(N(C(=O)CCOCCCOC)C)C1)C(C)C 30799,O=C(CC1=CCOCC1)NCCCCC1(NC(=O)CN2CCOCC2=O)CC1 30800,N1(C(C2C(C)CCC2)=O)CC2(CC2)CC1CNC(=O)Cn1cncn1 30801,CC1(C(=O)NCCOCCNC(C2CCCCNC2=O)=O)CCCNC1=O 30802,C1(CNC(CCCOCCOC)=O)Cc2ccccc2CN1C(c1cc[nH]c1)=O 30803,C(=O)CCCCCCCC=C.C#CCC(COC)OC(C)=O 30804,c1(CCN)cc(C(N2CC(F)(c3cccnc3)C2)=O)no1 30805,C(=O)(C1=NNC(C(F)(F)F)C1)N1CC(C)(NC(C(C(C)O)C)=O)C1 30806,c1(NC(CNC(=O)OCC)=O)ccc2c(COc3ccccc3)ncn2c1 30807,C(=O)(C1c2ccccc2CN1C(c1cnc(O)c(Cl)c1)=O)NC1CC(=O)NC1 30808,Cc1nc(C(N2CCC(CC(N3CCC(C(C)(C)O)C3)=O)C2)=O)c(C)s1 30809,C1(N(C)C(=O)C2CC2)CCN(C(=O)C#N)CCC1CO.N 30810,c1(C(N(C)CC2(O)CCN(C(C(CCOC)(C)C)=O)C2)=O)nn(C)c2c1CCC2 30811,c1(C(=O)NCC(CNC(CC(CC)CC)=O)OC)ccc(F)c2ccoc12 30812,CCCC(CCCNC(c1ccc(C(C)(C)C)cc1)=O)NCCCO 30813,C1(C(N2CC(C)CC(CC)C2)=O)(CC)CCCN(C(=O)CC#N)C1 30814,C1(C(=O)Nc2ccc(OC)c(N3CCOC3=O)c2)CCC(C2CC2)CC1 30815,N1(C(=O)NCN2CCC(C)(C)C2)CCC(CCC(=O)O)C(Cc2ccccc2)C1 30816,N1(C(C(C(C)C)SCC)=O)CC(NC(c2cnnn2C(C)C)=O)CC1(C)C 30817,c1(C(=O)NCC2C(C)(C)N(C(=O)CC3CC3)CC2)cc(F)c(O)c(F)c1 30818,c1(C(=O)NCC(C)CNC(c2ccnc3ccnn23)=O)cc2c(s1)CCCCC2 30819,c1(NCC2OCC(CNC(CSc3cn(C)nc3)=O)C2)ccnc2ncnn12 30820,C(CC(F)F)(C(=O)NC1CC2(CCCC2)C1)N(C(c1c(CC)con1)=O)C 30821,c1(C(C)C)[nH]nc2cncc(C(N3CCC(C)(NC(=O)C=CCO)C3)=O)c12 30822,c1(OC)cccc(C(N2CCCC(F)(F)C2)C(=O)NCC(C)C)c1C 30823,c1(NCCC2(O)CN(C(C(CC)SC)=O)C2)ncc(Br)cc1[N+](=O)[O-] 30824,C1(C)(C(=O)NCCCN(C(=O)CC2(C#N)CC2)C)CCC(=O)N1 30825,CC1(C2CC2C(=O)NCC=CC(=O)Nc2cncc(N(C)C)c2)COC1 30826,NS(=O)(=O)N1CCCC(C(=O)NC2(C3CN(C(=O)CCC(N)=O)C3)CC2)C1 30827,NS(=O)(=O)c1ccc(O)c(C(=O)NC2CC(NC(c3ccc(O)nn3)=O)C2)c1 30828,C1(NC(CCC(=O)NCCC)=O)CN(CCOCC)CCC1C 30829,C1(CC(=O)NCc2cn(CCNC(C=CSC)=O)nn2)CC2(CC2)CO1 30830,C1(C(N(CCCSC)C)=O)CCN(C(=O)C(C)c2cccs2)C1C(C)C 30831,C(c1ccc(F)cc1)=CC(N1CCN(c2nccc(CC#N)n2)CC1)=O 30832,S(=O)(=O)(c1cnccc1N1C2CCCC1COC2)NCC(c1cnn(C)c1)OC 30833,CC1(C)CC=C(C(=O)N2CCC3(CCCN3C(c3nc(Cl)ccc3N)=O)C2)CC1 30834,C(CC(C)(C)C(=O)N1CCN(C)C(C2CC2)C1)NC(C(C)n1cccc1)=O 30835,CCC(C(=O)N(C1(C(N2CCC3CCC23)=O)CCC1)C1CC1)C(F)(F)F 30836,N1(CCCNC(C(CC)C)=O)CCN(C(=O)C=CC(N2CCC(C)CC2)=O)CC1 30837,Cc1[nH]nc(C(N2CC(F)CC2CNC(=O)CCc2c(C)noc2C)=O)c1C 30838,C1(C)(CC)CCCN(C(C2CCC(O)CN2C(=O)CC2CCOC2=O)=O)C1 30839,N(C(=NCCC(C)C)NCCc1cnccn1)CC1(OC)CCC1 30840,C(=O)(CS(=O)(=O)C1CCCC1)N1CC(CN(c2cc3nncn3cn2)C)OCC1 30841,c1(C(N2CCOC(CCNC(C3CC(C(F)F)C3)=O)C2)=O)ccc2nnnn2c1 30842,C1(NC(C=C(CC)CC)=O)CN(C(=O)C(c2cccc(C)c2)(F)F)CC1O 30843,C1(CNC(C(CC)OCC)=O)CC(NC(=O)Cc2cscn2)C(O)C1 30844,C=CC1(CO)CCN(C(=O)C(C)(CSC)NC(=O)COc2cccnc2)CC1 30845,Cn1cc(CC(O)C(=O)NCCCOCCNC(=O)C=Cc2cnc[nH]2)cn1 30846,C1(C(=O)NCCC(CC)C)CC12CC(NC(c1cnccc1C)=O)C2 30847,c1(C(=O)NC(C2CCN(C(=O)C(F)=C3CCC3)CC2)C)ccc(N)cc1[N+](=O)[O-] 30848,c1nnn2c1CN(c1nc(N3CCN(C4CCOC4)CC3)nc(C3CC3)n1)CC2 30849,C(=O)(N=c1nc2ncc(Cl)cn2[nH]1)Cc1ncc(C(C)(C)C)o1 30850,n1(CC)nc(C)c(CC(N2CCOC(C(C)NC(=O)CCCN=[N+]=[N-])C2)=O)c1C 30851,N1(C(C2CCC(C)(C)OC2)=O)CCC(C2CC2)(CNC(=O)COCC(F)(F)F)C1 30852,Cn1c(=O)oc2c(C(=O)NCC(CNC(c3ccnc(O)c3)=O)CO)cccc12 30853,OCC1CN(CC2CC3(CCC(F)(F)CC3)C2)Cc2ccccc21 30854,N1(C(C(C)n2cnnn2)=O)CC(CNC(=O)Cc2ccsc2)CC(C)(C)C1 30855,N1(C(C(COCC)C)=O)CC2(CCN(C(=O)C(C)(C)c3cccs3)CC2)CC1C 30856,c1(C(N(C(CNC(c2cc(CC)c(CC)o2)=O)C)C)=O)ccn2cncc2c1 30857,N1(CC2CCN2c2c(C)cns2)CCC(c2n[nH]c(CNC(=O)C(C)C(C)C)n2)CC1 30858,c1(CCC(N2C(CN(C(=O)C(=Cc3c[nH]cn3)F)C)CCC2)=O)cccc(F)c1 30859,N1(C(c2cc(CCC)on2)=O)CCC(O)(CN(C)C(C2CCN(C)C2=O)=O)C1 30860,C1(C(=O)Nc2cc(Br)cc(OC)n2)COC2(CCN(C(=O)CCC(C)C)CC2)C1 30861,N1(S(CC=C)(=O)=O)CCCN(C(c2ccc(Cl)cc2F)=O)C(C)C1 30862,S(=O)(=O)(C(F)(F)F)N1CC2C(C(N3CCOC(C4CCC4)C3)=O)C2C1 30863,N1(C(CC(C)n2ccnc2)=O)CCC2(CC1)CC2NC(C1(C(F)(F)F)CC1)=O 30864,c1(C(N2CC(O)(CNC(C3(C)C(CC)CCC3)=O)C2)=O)ccc2oc(=N)[nH]c2c1 30865,C12(NC(Cc3cc(CC)no3)=O)CCCCCC1N(C(c1nnsc1N)=O)CC2 30866,CC#CCCC(=O)N1CCC(C(N2CCC2C(=O)OC)=O)O1 30867,N1(C(=O)CCN(C(c2ccco2)=O)CC2CC2)CC2(CCC2O)C1 30868,n1(CCCC)nnnc1C(c1csnc1OC)NCC(n1cccn1)C 30869,CCCCCCC(=O)NC1(CC(N2CCC3CC2C(=O)O3)=O)CCC1 30870,c1(C(=O)NC(C)CN(C(=O)CC2CCOC2)C)cc(C(F)(F)F)ncc1N 30871,C(=O)(CCS(N)(=O)=O)NCC(C(C)(C)C)NC(CCC(C)SC)=O 30872,c1(CC(C(=O)N(CCNC(=O)Cc2cc(C)[nH]n2)CC)O)ccccc1Cl 30873,C(C(=O)NC(C)CCSCCOC)(C(C)C)NC(CCOCCC)=O 30874,C1(CNC(C(C)(C)CC=C)c2n(CCOC)nnn2)COc2ccccc2C1 30875,C1(C(C#C)NC(=O)N(CCCN(C)C)C)CC(F)(F)C1 30876,S(=O)(=O)(c1cc(F)c(OC)cc1C(=O)OC)NC(c1c(OC)scc1)=O 30877,C1(CNC(c2c(CC)ccs2)=O)CCCCC1NC(c1cc(OC)n(C)n1)=O 30878,c1(N2CCC(Nc3c(C(=O)OC)c(C)sc3)C2=O)cc2ccccc2o1 30879,Cc1ccn(C)c1C(=O)NCCC1CCCN(C(C2(O)CCCCC2)=O)C1 30880,N1(C(c2ccnnc2CO)=O)CCCS(=O)(=O)CC1C1CC1 30881,C(=O)(C(O)C(C(C)C)OC)NCCC(CNC(C(F)=CCC)=O)(C)C 30882,c1(CNC(N2CCC(CN)C2c2cccnc2)=O)cc(Cl)c(F)c(Cl)c1.C1C(=O)N1 30883,c1(OC)ccc2c(c1)C(C(=O)NCC1C(NC(c3ccoc3C3CC3)=O)C1)CC2 30884,C1(C(=O)NCC2(C)CCN(C(C=COCC)=O)C2)CCC12CCOCC2 30885,N1(C(c2cn(CCCOC)nc2)=O)CC(NC(c2ccoc2Br)=O)C(O)C1 30886,c1(C(=O)NC2C(C)CN(C(c3nn(C)cc3Cl)=O)CC2)cc2c(cc1O)OCO2 30887,N1(C(C(C#C)(C)C)=O)CC2CC(NC(=O)CCc3cncc(O)c3)C(C2)C1 30888,c1(NC(C(COCC)NC(=O)CC2CC2(C)C)=O)ccn2nccc2c1 30889,c1(C(=O)NC(CCN(C(c2ccc(SC)o2)=O)C)C(C)C)c(C)ccc(C)c1N 30890,C1(C(=O)NC(C2(C(N3CCC3CC(N)=O)=O)CC2)C)CC=CC(O)C1 30891,C12(CNC(c3cc(CO)ccc3Cl)=O)CCC(CC1)CN2C(=O)C(F)F 30892,CC1CCN(C(c2cc(C(F)(F)F)cs2)=O)CCN1c1ncc(I)cn1 30893,Cc1nn(-c2cccc(F)c2)cc1C(N1CCCC(NCC(F)F)C1)=O 30894,c1(C(=O)NC2CC(C)N(C(=O)C3=CCOCC3)C2)c[nH]c(=N)nc1O 30895,Cc1cnncc1C(=O)NC1(C)CC(NC(C2CCCSC2)=O)C1 30896,N1(C(C(C)OCCCCCC)=O)CC(NC(c2ccnnc2C)=O)CC(C)(C)C1 30897,N1(C(C=CCC)=O)CC(O)(C2(CNC(c3c(C)cc(F)cc3Br)=O)CC2)C1 30898,C1(CNC(C(CN(C)C)(F)F)=O)CC2CCC1N2C(C1(C2CCCO2)CCC1)=O 30899,CCCCCC(O)C(=O)NCC1CN(C(c2cnc(N(C)C)o2)=O)CC12CCC2 30900,n1(COC)ccc(C(=O)NCCCOCCC(=O)NCCc2noc(C)n2)n1 30901,C1(CNC(C(CC)=CCCC)=O)CN(C(=O)COC)CCN1C 30902,N1(C(C(C)CC(C)(F)F)=O)CCOC2(C1)CN(C(=O)CCCC1CCOCC1)C2 30903,C=CCCC(CO)NC(=O)C(O)C1CN(C(c2cn(C3CC3)nn2)=O)C1 30904,c1(NC(C2(C)CCN2C(c2ccc3nc[nH]c3c2)=O)=O)ccc(Cl)c(C#N)c1Cl 30905,n1(C(C)C(N2CCC(F)(CNC(=O)CCNC(N)=O)C2)=O)cc2ccccc2n1 30906,C(c1ccncc1)=C(C(=O)NC(CCN(C(C(CC)F)=O)C)C)C 30907,c1(CNC(c2ccc(-c3ccc(SC(C)C)cc3)cn2)=O)c(O)ccc(F)c1F 30908,C(=O)(C(CO)NC(c1[nH]ccc1C)=O)OC.C12CC(C1)NC2=O 30909,C1(c2cnccc2)CCN(C(=NCC2CCC(N3CCCCC3)CC2)NC2CC2)C1 30910,c1(C(C(C(=O)Nc2ccc(C(c3n(C)ccn3)O)cc2)N)=O)ccc(F)cc1F 30911,C1(CC#C)(NC(=O)C(C2CN(C(C3CC4CC4C3)=O)C2)OC)CC(CO)C1 30912,c1(OC)cc(C)c(Br)cc1C(N1CCC2(CC1)CC2NC(c1cc(C)[nH]n1)=O)=O 30913,N1(C(CC2CC(=C)C2)=O)CCN(C)CC1C(=O)NCC(CC(C)C)N(C)C 30914,CON(C)C(=O)CNC(C1(CNC(=O)C(c2ccn(C)n2)C)CC(C)(C)C1)=O 30915,C(CC(=O)N1CCC(OCCF)C1)(C(F)(F)F)NC(C1C(C)(C)C1(F)F)=O 30916,N1(C(C2C(CC)CCC2)=O)CCC(C(=O)NCC2(N(C)C)CC2)(CC)CC1 30917,c1(-c2ccc(SCC)cc2)ccn2nc(C(=O)NCC#N)cc2c1.C1(O)CCC1 30918,C=C1CCN(C(=O)C(C)OC2CCCC2)C(C(=O)NCC(C2CC(C)(C)C2)O)C1 30919,Cc1nc2c(s1)CCCC2C(=O)NCC1(CNC(=O)C(C)SC(F)(F)F)CC1 30920,c1(OCC)oc(C)nc1C(=O)NCC(CCNC(=O)CCC(C)SC)OC 30921,C1(C(N2CCC(N=[N+]=[N-])C(O)C2)=O)CC12CCOc1ccc(F)cc12 30922,N1(c2cc(N(CCC3CN(C)C3)C)ncn2)CCCC2(CCCCCC2)C1 30923,C(CCC1CCC1)(C(=O)NCc1cnn(C)c1O)NC(c1c(C)ocn1)=O 30924,c1(C(=O)NCC(CC)NC(=O)C(C2CCCCC2)F)ccc2nnnn2c1 30925,c1(C(=O)NC2CC(N(C(CCC(=O)NC)=O)C)C2)cc(N)nc(Br)c1 30926,C(C(=O)N(CC)OC)NC(C(CNC(C1(CC#C)CCC1)=O)C)=O 30927,N1(C(c2c(C)nsc2N)=O)CC(C2CN(C(=O)CCC3CCCOC3)C2)C1 30928,N1(C(C2CNC(=O)N2)=O)CCCC2(CCN(C(c3cocc3C(N)=O)=O)C2)C1 30929,C(=O)(C1CCc2cccc(F)c21)NC(CC)CNC(=O)Cn1ccc(=O)cc1C 30930,C=CC1(C(=O)NC2CCCCC23CC3)CCN(C(=O)Cc2cscn2)C1 30931,CCC(C)CCCCC(=O)NCC(CC)N(C(=O)Cn1cc(C)cn1)C 30932,N1(C(c2ccn(CCC)n2)=O)CC2CCC(C1)N2C(c1cnc(C2CC2)s1)=O 30933,c1(C(=O)NC2CCC(CCNC(C(C(C)C)C)=O)C2)nn(C)c(Cl)c1Br 30934,N1(C(C(CC)OCC2CC(C)CC2)=O)CC(OC)CC(NC(=O)C2CC2)C1 30935,C(=O)(C(COC)COC)NCC1(C(=O)NCC2C(CC)C2)CCC1 30936,C(=O)(C(CC(C)C)NC)NCc1nc(-c2scc(C)n2)nn1-c1cccc(F)c1 30937,C1(CN(C(=O)CN(C)C(C2(C)COCCO2)=O)C)CCCCCC1 30938,c1(C(=O)NCC(C2CCCCC2)NC(C(C(C)C)F)=O)csc([N+](=O)[O-])c1 30939,C1(NC(C(CC)=CCCC)=O)CCN(C(=O)COc2cc(C)on2)CC1F 30940,C(C(=O)OC)(C(C)(O)C(F)F)N1CC(C(=C)C)OCC1 30941,N(C(=NCCc1cnc(C)cn1)N1CCC(CS(C)(=O)=O)C1)CC(=C)C 30942,C1(CNC(CCOC)=O)CN(C(C23CC(F)C2C3)=O)CC12CCOCC2 30943,N1(C(c2cccc(OCC#N)c2)C(=O)NC)CCOc2cccc(Br)c2C1 30944,C(=O)(C(C)(CC)CC)NC(CNC(Cc1c(SCC)cccc1)=O)CCOC 30945,c1(NC2CCC(C(=O)Nc3cnc(C)nc3Cl)CC2)nccc(S(C)(=O)=O)n1 30946,c1(N2CC(C)C(NC(c3cnsn3)=O)C2)ncc([N+](=O)[O-])cc1Cl 30947,c1(C(=O)NC23C(n4cc(C(CC)O)nn4)CC(CC2)C3)cccc2c1SCCC2 30948,N1(CC)CCCC1(C(=O)NCC1CC1N(C)C)CC.c12cc([nH]n1)CNC2=O 30949,c1(N(C=O)C)ccc(Br)c(Cl)c1 30950,N1(C(C(CC)c2ccccc2)=O)CCN(C(c2n[nH]c(C)c2F)=O)C2(CCC2)C1 30951,N1(C(C2CC(CC)C2)=O)CCc2cc(NS(=O)(=O)c3cccc(Cl)n3)ccc2C1 30952,CC1CCC(NC(c2c[nH]ccc2=N)=O)CN1C(c1csc(-c2cccs2)n1)=O 30953,C1(NC(CC(C=C)CCC)=O)CCC2(CCCN(C(=O)C3=C(Cl)CCOC3)C2)C1 30954,CC1CN(C(=O)C(C)Cn2cccn2)C(C)C1C.C123COC(C1)C(C2)NC3=O 30955,c1(C(N2CCC(NC(Cc3c(C)con3)=O)(CO)C2)=O)c(C)cccc1[N+](=O)[O-] 30956,C(O)(CN=C(NCC(F)F)NCC1(C)CC1(F)F)c1cc(C)cc(C)c1 30957,N1(C(CCCC(C)=O)=O)CC2CCCN(C(C3OCCN(C)C3=O)=O)C2C1 30958,N1(C(c2c(OC)nsc2)=O)CC(CC(=O)NCC2CC2C(C)C)C2(CC2)C1 30959,c1(CC)cc(C(=O)NCCCCCNC(=O)C(CC)n2nccc2C)c(C)nn1 30960,C1(NC(CC=C)=O)CCN(C)C12CCCN(C(C1CCCN1C1CCCC1)=O)C2 30961,c1(C(=O)NC2CN(C(c3cc(OC)cc(F)c3)=O)CC2F)cc(Cl)c(F)cc1F 30962,n1(CC)cc(C(=O)NCC2CCC(NC(C3CNC(=O)N3)=O)C2)c2ccccc12 30963,N1(C(C(CC#C)C)=O)CCc2ccccc2C(NC(=O)C(C)(C)C(F)F)C1 30964,N1(C(c2c(CC)nnc(C)c2)=O)CC2(CCN(C(C3(C(N)=O)CCC3)=O)CC2)C1 30965,c1(NC2CCCC(NC(C=Cc3c(C)n(C)nc3)=O)C2)ncc(C#N)cc1Br 30966,C(=O)(CCN(OC)C(=O)CC1CNC(=O)O1)NC(CCCC)CCC 30967,c1(OC)cc(C(=O)NCC2CCCCN2C(c2nccn2C)=O)ccc1O 30968,C1(C)(CNC(C2(N(C(C(CN(C)C)O)=O)C)CC2)=O)CC2(CC2)C1 30969,C(CC(=O)CNC(=O)NC(CC(=O)OC(C)(C)C)(C)C1CCC1)C1C(C)C1 30970,Cc1ccc(F)c(OC(=O)Cc2cccc(NC(c3cc(C)cc(Cl)c3)=O)c2)c1 30971,N1(C(CN(C)CC)=O)CCC2C(CCCN2C(c2cc3nc[nH]c3cn2)=O)C1 30972,N1(C(C(CSC)C)=O)C2CCC1CC(C(N1CCC(F)(CO)C1)=O)C2 30973,c1(C(=O)NCCC(C)NC(=O)CCc2nc(O)n[nH]2)c(F)ccc(F)c1N 30974,C1(C(N2CCC(CNC(CCSCC(N)=O)=O)C2)=O)COc2cc(Cl)ccc2C1 30975,C1(C(=O)NCCN(C(=O)CN(C)C2CC2)CC)CCCC1O 30976,N1(C(C(C)(C)C2CCC2)=O)CCC(NC(=O)CC=CC(=O)O)CC1 30977,CCC(CC(=O)NC(CCN(C(=O)C(C)Cc1ccccc1C)C)C(C)C)SC 30978,c1(C(N2CCCC(NC(COCCOCC)=O)C2)=O)ccc(O)cc1C 30979,c1(SC)cccc(C(=O)NC2(C)CCN(C(=O)C(C)(C)CC(F)F)C2)c1[N+](=O)[O-] 30980,N1(C(CCSCC)=O)CCC2(CC1)CC2(CO)CNC(C1CC1c1cccs1)=O 30981,CC1(C)CC(CNC(c2cncc(Cl)n2)=O)N(C(=O)C(C2COC(C)(C)O2)O)C1 30982,c1(C(=O)NC(C2CCCCN2C(=O)Cc2cocn2)C)nn(C)c2c1COCC2 30983,C(=O)(C(C)(F)C(=O)NC1CC(CNC(c2cc(Cl)cc(Cl)c2)=O)C1)OC 30984,N1(C(CNC=O)=O)CCN(C(C2CCCC23CCC3)=O)C2CCC12 30985,C(C1=CCN(C(C2CCC3CC3C2)=O)CC1)NC(c1ccnn1CC1CCC1)=O 30986,C1(NC(c2ccsc2Cl)=O)CN(C(=O)C(F)=CC2CC2)CC12CCOCC2 30987,N1(C(=O)COCCF)CCN(C(C23CCCC2C3)=O)C2(CC2)C1 30988,C1(CNC(C(N)=O)=O)CC(NC(=O)Cc2cccc(OCC(F)F)c2)C12CCC2 30989,c1(C(N2C3(CNC(CC(CC)O)=O)CC(C2)C3)=O)cc2cc(C)cc(C)c2[nH]1 30990,C(CS(=O)(=O)CC(=O)NC1CC1CNC(c1nc(C)c(C)nc1C)=O)OC 30991,N1(C(C(C)(C)SC)=O)CCC(NC(=O)CCc2cocn2)C2(CCC2)C1 30992,c1(C(=O)NC2C(NC(C(CC(C)C)NC(C)=O)=O)CC2)cc2ncccc2s1 30993,Cc1ccc(F)c(C(=O)NC(C2CCN(C(=O)CC3NC(=O)NC3=O)CC2)C)n1 30994,N1(C(c2cc(C)cc(F)c2)=O)CC(C)CN(C(C2COC3COCC23)=O)CC1C 30995,CC1CCCCCC1NC(=O)C=CC1CCCN1C(=O)CC1CCSCC1 30996,N1(C(C(CC=CC)NC(=O)C=CC(C)(C)SC)=O)CCC2(C=CCO2)CC1 30997,C=C(CNC(c1cc(C)c(I)s1)=O)c1ccc(C)c([N+](=O)[O-])c1 30998,C12(CC(=O)NCCNC(c3c(CCC)onc3C)=O)CC3CC(CC(C3)C1)C2 30999,Cc1ccc(C(=O)NC(C)(C)CNC(=O)CC2CC(O)C2(C)C)c(F)c1Br 31000,CC1CC(NC2CN(Cc3ccccc3)CCC2O)C(=O)N1c1ccccc1 31001,C#Cc1cc(C(=O)NCC2CCC2NC(=O)Cc2sc(C)cc2C)cc(N)c1 31002,N1(C(c2cccc(OC)c2O)=O)CCC2CN(C(C3CCCC(C)C3)=O)CC2C1 31003,c1(CNC(C2(C=C)CCC2)=O)ncc(C(N2CC(OC(=O)N(C)C)C2)=O)cn1 31004,c1(C(N(CC=CC(=O)N(C2(COC)CC2)C)C)=O)ccc([N+](=O)[O-])o1 31005,C(C)(C)(C(=O)NCCC(C)(C)NC(=O)C(C)Sc1nnnn1C1CC1)OC(C)=O 31006,c1(C(N2CC(C)C(NC(=O)C(c3ccc(F)c(F)c3)O)C2)=O)nc(Cl)ccc1N 31007,O=C(C1CCCc2nccn21)NCCNC(=O)CC12CNC(=O)C(C1)C2 31008,N1(C(C(CC=C)N(C)C)=O)CCC(C2CC2)C1CNC(=O)Cc1ccc(F)cc1 31009,c1(C(=O)NC2C(NC(C(CC)(C)O)=O)C2)c(SC)cccc1F 31010,c1(C(=O)NCCC2(C)CCN(C(C3(SC)CC3)=O)C2)cc2n(n1)CC(C)NC2=O 31011,CC1CN(C(C2C3(CC3)C23CC3)=O)CC2(CCN(C(=O)CC3OCCO3)C2)O1 31012,N1(C(CSCC#C)=O)CCC2(CC1)CN(C(=O)Cc1nonc1C)C2 31013,C12(C(N3CCCC(CNC)C3)=O)CCC(C(F)(F)F)(C1)OC2 31014,C12(NC(COCc3cn(C)nc3)=O)CCC(CC1NC(=O)CSc1ccsc1)C2 31015,N1(C(C2CC(=O)C2)=O)CCC2(C=C(C(=O)NOCC(F)(F)F)C2)C1 31016,CCCC(C)=CC(=O)NC(C(=O)NCC(O)COCC)C1CCC1 31017,c1(C(=O)Nc2ncc(F)cc2F)nc(=NCc2ccccc2)[nH]cc1Cl 31018,C1(NC(C2(Br)C(C)(C)C2)=O)CCCN(C(c2ccc(F)o2)=O)CC1 31019,c1(C(=O)NCCCC(CO)NC(CCc2cnc(C)s2)=O)cccc2nccn12 31020,Cc1cc(C(=O)NCC(C)NC(=O)COc2cccc(O)c2)ccc1F 31021,C(CCCCCCC)NC(C1CCCN1C(C1(NC(C(C=C)(C)O)=O)CC1)=O)=O 31022,c1(CNC(C(c2cnccn2)C)=O)ocnc1-c1cn(C(c2nncs2)C)nn1 31023,C(=O)(C(=O)CCC(C)C)NC1CCN(CC(=O)Nc2c(SC)cc(C)cc2)C1 31024,N1(C(c2cc(CC)on2)=O)CC(NC(c2coc(Cl)n2)=O)Cc2ccccc21 31025,N1(C(c2cnc(OCC)s2)=O)CC(C)CN(C(c2oc(C)nc2C)=O)C(C)C1 31026,c1(CCNC(=O)C(=O)NCC2(F)CC3(CNC3)C2)ccc(Br)cc1Cl 31027,N1(C(CC(C)SC)=O)CCCCC1CCCNC(=O)CCCc1nc(C)cs1 31028,CC1(C)CC(CO)CN1C(C1CCCN(C(=O)CCC2CCOC2)CC1)=O 31029,C(c1cc(C(F)(F)F)ccc1Cl)=CC(N1CC(CNC(=O)CCF)OCCC1)=O 31030,C#Cc1cc(C(=O)NC2(CNC(=O)C(F)(CC)C(=O)OCC)CCC2)ccc1Cl 31031,CC12CCN(c3ccncc3C#N)CC1C2(Cl)Cl 31032,C1(NC(C(C2CCN(C(CC3CC(=C)C3)=O)C2)F)=O)CCCCC1(C)O 31033,n1(CC)nc(C(=O)NC(C)CC(C)NC(=O)C(c2ccc(F)cc2)=O)c(C)n1 31034,C1(C(N(C2CC(C#N)C2)CC(=O)NCCc2c(C)ocn2)=O)CC(=O)NC(C)C1 31035,Cc1cc2[nH]c(=O)c(C(=O)NCCC3CN(C(C4(Cl)CC4)=O)CC3C)cn2n1 31036,Cn1c(C2CC2)nn(CC(=O)NC2CCC2CNC(=O)Cn2cnnc2O)c1=O 31037,N1(C(c2cccc(CCC)c2)=O)CCCC(F)(C(=O)NCc2cnsc2)C1 31038,O(NC(=O)C(F)(CNC(=O)CCC(F)(F)F)C(C)C)CC#C 31039,C(C(=O)N=c1cc(C)o[nH]1)SCC(=O)NCCCC(CO)NC(CCCC=C)=O 31040,N1(C(CC(C)OC)=O)CC(CCNC(=O)CCc2cncc(Br)c2)C(C)C1 31041,CCCC(C(O)c1ccccc1)NC(c1sccc1Cl)COC 31042,C(C(C(=O)N1CC(C)(CSC)C1)C(C)(C)C)NC(C=CC(CC)C)=O 31043,C1(C)(C(N2CCN(CCCNC(c3c(C)ncnc3)=O)CC2)=O)CCCCC1C 31044,CC(C(C(=O)NC1(C)CC1)N1CCC(O)(C(N)=O)C1)C1CCC1 31045,Cc1ccc(S(=O)(=O)NC2CN(C(c3cccc(C)c3Cl)=O)CC2F)c(F)c1 31046,c1(C2C(NC(=O)NCCc3cc(OC)ncc3)C2)cc(C)cc(Br)c1 31047,CCCC(C)CCCC(=O)NC(CNC(c1ncc(OC)cn1)=O)C(C)(C)C 31048,S(=O)(=O)(CCC(=O)NC1CCC(NC(=O)C(CO)N(C)C)C1)NCCNC(C)=O 31049,C1(C)(NC(COc2ccc(C(=O)OC)cc2)=O)CC(CC(=O)NC(C)C)CC1 31050,N1(C(C#C)=O)CCCC(C(=O)Nc2c(C(N)=O)cccc2C)CC1 31051,N1(C(c2c(C)nn(C)c2Cl)=O)CC2(CCN(C(=O)CCc3cncc(O)c3)C2)C1 31052,C1(CSC)COCCN1C(=O)C(n1cc(COC(=N)O)nn1)C 31053,c1(C(N(C2CCCN(C(=O)C(C)=C3CC3)CC2)CC)=O)ncc(OC)cc1F 31054,O=C(N=c1c(Cl)c[nH]cc1I)C1CC12CCN(C(c1ccccc1Br)=O)CC2 31055,N1(c2cc(C)nc(Cl)n2)CCCC(C2CCN(C(=O)C(C)(C)S(C)(=O)=O)CC2)C1 31056,CC(CC(=O)N1CCN(C(=O)CCc2ccc[nH]2)C(CCO)C1)C(F)(F)F 31057,c1(C(N2CCOC(CCOC)C2)C(=O)NCCC(=O)OCC)cc(C)nc(C)n1 31058,CC1C(NC(c2cc(F)ccc2F)=O)CCCN1Cc1cnon1 31059,N1(C(C2ON=C(C)C2)=O)CCCN(C(c2cccc(=O)n2C)=O)C(C)C1 31060,c1(C(N2C(CN(C(C(C)OCCC(C)C)=O)C)CCC2)=O)ccccc1C(C)O 31061,C(=O)(CCCC(=O)N1CCC(CNC(c2ncoc2C)=O)C1)OCC 31062,N1(C(C(CC)CC)=O)CCCC(NC(C23CCN(CC2)CC3)=O)CC1 31063,c1(C(N(CC(CC)NC(c2cc(OC)ccc2O)=O)C)=O)cnn2cnnc2c1 31064,N1(C(C=CCN(C)CC)=O)CC(OC)CC(NC(=O)CC2CC(OC(C)(C)C)C2)C1 31065,C12(C(N3CCC(CC(=O)NCC4CCCOCC4)C3)=O)CCC(CO)(CC1)C2 31066,c1(OC)c(C(N2CC(CO)(NC(c3ccc(=O)oc3)=O)C2)=O)cnn1C 31067,Cc1c(C(=O)NC2(CNC(C3CC4(C3)CC4(F)F)=O)CCCCC2)cncc1F 31068,n1(CC(=O)NC)ccc2ccc(NC(=O)C(N3CCC(CO)(CO)C3)=O)cc12 31069,n1(CCNC(=O)CNC(C2CCCC2)=O)cc(-c2nccs2)nn1 31070,CN1CCN2CCN(C(c3cnn(-c4cccc(Br)c4)n3)=O)CC2C1=O 31071,N1(C(c2c(CC)cccc2F)=O)CCCC1C1CCCN1C(c1ccc(Cl)o1)=O 31072,C(CN=c1ccc(S(=O)(=O)NC2CCCCC2O)c[nH]1)SCC(C)C 31073,CC1(C)CCN(C(C2CC2(C)C)=O)C(C(=O)Nc2ccc(F)c(O)c2)C1 31074,c1(CC(=O)N(CCCNC(CC2C(CC)C2)=O)CC)ccc(OC)c([N+](=O)[O-])c1 31075,C1(N(C(CCOCCN(C)C(C2CC(=C3CC3)C2)=O)=O)C)CCSCC1 31076,c1(C(CNC(=O)CC2CC2CSc2ccccc2)OC)ncc(C)s1 31077,CC(CCCNC(C1(C2CCCO2)CCCC1)=O)NC(c1ccon1)=O 31078,CC1CN(C(C2CCCC2F)=O)CC(C)CN1C(c1cnn(C)c(=O)c1)=O 31079,C1(NCCCC2(NC(C(C)NC(CC)=O)=O)CC2)CC(OC)C(OC)C1 31080,N1(C(c2c(C#C)c[nH]n2)=O)CCCC(COC)(NC(C2CCCN2C2CC2)=O)C1 31081,C(=O)(C(C(=O)N1CCCC(CC(N2CCC(C)(N(C)C)C2)=O)C1)OC)OC 31082,C1(NC(CNC(CC(C)C)=O)=O)CCC(C)N(C(=O)C=C2CCOCC2)C1 31083,C1(CNC(c2n(C(C)(C)C)ncc2)=O)CCCC(NC(C2C3CCCC23)=O)C1 31084,C1(CNC(C(COC)O)=O)CCN(C(C2CC(c3cccc(F)c3)C2)=O)C1(C)C 31085,N1(C(C2C(NCc3ccc(COC(C)=O)o3)C2)=O)CCc2cccnc2C1 31086,c1(C(=O)NC(C(=O)NC(CN(C(CCOC(C)C)=O)C)C)C)ccccc1Cl 31087,C(=O)(C1CCc2c(Cl)cccc21)N1CCCC(C)(C)C1CNC(=O)COC1COC1 31088,CC1=NOC(=O)C1CC(N1CCOC(CN(C)C(C2CN(C)CCO2)=O)C1)=O 31089,c1(NCCOC(C)=O)ccc(C(N2CCN(c3ncco3)CC2)=O)cc1C 31090,Cc1ccc2c(C(=O)NC3(CCNC(=O)CC(C)P(C)(C)=O)CC3)onc2c1 31091,N1(C(=O)CCc2ccon2)CCC2CN(C(=O)CCc3ccc(CO)cc3)C2C1 31092,C(C)(C(=O)NCC(C)N(C(=O)CNS(=O)(=O)N(C)C)C)(C(C)C)OC 31093,N1(C(CNC(C)=O)=O)CCC(C)(C(=O)NC(c2cccc(OC(F)F)c2)C)C1 31094,c1(CC(=O)N(C)CC2CCCN(C(=O)CS(C)(=O)=O)C2)cnc2cccnn12 31095,C#CCC(C)(C(=O)NC1CN(C)NC1=O)NC(C1CCCCN1C)=O 31096,C1(C)(C(=O)NCC(N(C(Cc2nc(CC)sc2)=O)C)C2CC2)COC(=O)C1 31097,Cc1ccc(N)c(C(N2CCCC2C(C)NC(=O)Cc2cccnc2)=O)c1 31098,C1(CCC(=O)NC)CN(C(=O)N(C)CCOCCOC)CCC1C 31099,n1(CC)ncc(C(=O)NCC2(NC(C3(C)CCSCC3)=O)CC(OC)C2)c1C 31100,c1(C(=O)NCc2scc(CNC(c3cc(C)ns3)=O)n2)cc(O)nc(C2CC2)n1 31101,CC(C)C(O)C(C)C(=O)NCC1(F)CN(C(c2ncn3c2CCC3)=O)C1 31102,c1(C(N(CC(C)NC(C(C2CC(F)(F)C2)OC)=O)C)=O)coc(C#N)c1 31103,c1(C(C(=O)OCC)=O)c[nH]c(=NCC(C)NC(=O)CC2CCCC(C)C2)c(C)c1 31104,c1(C2C(C(F)(F)F)(C(=O)NC3(c4nc[nH]n4)CC3)C2)ccccc1-c1nn[nH]n1 31105,c1(CCC(=O)NC(CN(C)C(c2ccc(Cl)s2)=O)(C)C)ncc(F)cn1 31106,c1(OC)ccc(C(N2CCCC(NC(=O)C(F)(F)C(F)F)C2C)=O)c(N)c1F 31107,N1(C(Cc2ccc(OC)cc2F)=O)CCN(C(C2(C)CCOC2)=O)CC2(CC2)C1 31108,c1(CC)cc(C)[nH]c(=NC(C)CC(C)NC(=O)CN2Cc3ccccc3C2)n1 31109,c1(CC(=O)NCC(C)NC(C2(CS(C)(=O)=O)CC2)=O)ccc(OC(F)F)c(F)c1 31110,C(=O)(C1CCc2nccn21)N1CCN(C(CCC2C(C)C2)=O)CC1CO 31111,c1(NCC2CCN(C(=O)CSc3ccc(F)cc3)C2)ccc2c(c1)CCN2 31112,CC1=C(C(=O)N2CCCC2CCNC(c2ccc(F)c(F)c2F)=O)CCS1(=O)=O 31113,CC(CNC(C1CC1(C)C(F)F)=O)C(F)C(=O)NCC1CSC1 31114,C#Cc1ccc(C(=O)NC2(C(N3CCC(CO)C3(C)C)=O)CC(O)C2)nc1 31115,N1(C(C2C(CNC(c3ccsc3Cl)=O)CCC2)=O)CC(CO)C2(CCC2)C1 31116,C1(=O)C(F)CC(C)(C)N(C)CC2(CC)COCCN12.CCOC 31117,C1(C)(C(NOC2CCCN(CC)C2)=O)CC(O)CN1C(=O)CCc1cscn1 31118,C1(CNC(C2C(CCC)C2)=O)(CO)CC12CCN(C(c1cnnn1C)=O)CC2 31119,CC1(C)CC(C(N2CCOC(C#N)C2)=O)CN1C(C1CC2CC(=O)C1C2)=O 31120,c1(C(=O)NC2CN(C(C(COC)(C)OC)=O)CC2C)ccc(F)c(C(C)C)c1 31121,[N-]=[N+]=NC1CN(C(c2ccc3cc[nH]c3c2)=O)CC1NC(=O)COC(F)F 31122,C1(C)(C(N(C2CN(C(=O)Cc3cn(C)nc3C(N)=O)C2)C)=O)CCCS1(=O)=O 31123,N1(C(Cc2nnc(C)o2)=O)CCC(C2CC2)(NC(c2ccc(C)c(F)c2F)=O)C1 31124,N1(C2CN(C(C=CC(=O)N(C)C)=O)C2)CCN(C(C23CCCCC2C3)=O)CC1 31125,C(=O)(CCC(C)NC(=O)C(C)NC(N)=O)NC(c1nc(C)on1)C 31126,C(CN=c1[nH]c(=NCCc2cccn2C)[nH]c2cc(C)ccc12)NC(C)=O 31127,C=CC(CC)CC(=O)NCC1CN(C(C2CC3(CC(=O)N3)C2)=O)CCN1C 31128,c1(C(N2CCC(C(C)NC(C3(F)CCC3)=O)C2)=O)ccnc(NC2CCC2)c1 31129,C(C1(C)OCCc2ccccc21)NC(C)(C)CCc1ccc2c(c1)OCO2 31130,C1(C)(CNC(C(CSC)C)=O)CN(C(c2ccc(OC)nc2F)=O)C(C)(C)C1 31131,C1(NC(CC=CCC)=O)CCN(C(c2cncc(S(C)(=O)=O)c2)=O)CC12CCC2 31132,N1(C(C(C)c2cccs2)=O)CCCC(CCNC(=O)COc2ccccc2)C1 31133,N1(C(Cc2n(C)cnn2)=O)CC2CC(NC(c3ccnn3C3CCC3)=O)CC1C2 31134,N1(C(C2C(C)(Br)C2)=O)CCC2(CCN(C(c3cn(CC4CC4)nn3)=O)C2)C1 31135,Cc1nc(C(=O)NC2C3CN(C(=O)C=CC4CCC4)CC23)c(=O)[nH]c1C 31136,c1(C(=O)NCC(CC)NC(=O)Cc2cnccc2C)c(N)cc(Cl)nc1Cl 31137,C1(C(=O)OC)CCCC1C(=O)N(CCCN(C)C(C1CCSC1)=O)C 31138,C(=O)(CS(=O)(=O)CC(C)C)NC1CC2CC(NC(C(C(=C)C)(C)C)=O)CC2C1 31139,c1(C(=O)NC(CC)(C)CNC(C2(C)CCOCC2)=O)nc2ccccc2cc1C 31140,Cc1cc(C)c(OCC(=O)N(C2C3CN(C(C4(CCO)CC4)=O)CC23)C)c(C)c1 31141,C1(C(=O)Nc2cc(Cl)ccc2Br)COC2(CCN(Cc3ccc(Br)cn3)CC2)C1 31142,c1(C(N2CC(CCNC(C3(CC)CC3)=O)(OC)C2)=O)c(Cl)nn(C)c1Cl 31143,C1(NC(c2cc(OC)n[nH]2)=O)CC2CCC(C1)N2C(C1CCCC1C(C)C)=O 31144,N1(C(C(CC)C(C)O)=O)CC2(C1)CN(C(=O)CCCc1ccc(O)cc1)CCO2 31145,C1(NC(C(C)(C)C2CC2)=O)CN(C(C2CCC3(C2)N=N3)=O)CCC12CCC2 31146,CCCCCC(O)CC(=O)N1CCC(NC(c2c(Cl)ccc(F)c2F)=O)C(F)C1 31147,c1(C(C(=O)NCC2(C(=O)NC(c3cccs3)C)CC2)C)ccccc1 31148,C(C(F)(F)CCC(=O)NNC(=O)c1cnccn1)n1cc(CC(COC)O)nn1 31149,c1(CC(N2CC(CNC(CCOCCCC)=O)C2)=O)nc(C(C)OC)n[nH]1 31150,C12(CNC(=O)Cc3cc[nH]c3)CCCCC1CN(C(c1ccc(O)nc1Cl)=O)C2 31151,N1(C(CC=C)=O)CCCCC1CN(C)C(C1(n2cccn2)CCOCC1)=O 31152,C1(CNC(c2n[nH]c(C)c2C)=O)CN(C(C2CS(=O)(=O)C2)=O)CC1(F)CO 31153,C1(F)(C(=O)NCCCOCCNC(C(c2ccc(CC)s2)=O)=O)C2CCCCC12 31154,c1(C(=O)NCc2n(C)ncc2)ccc(C(=O)NCC2CNC(=O)CO2)cn1 31155,C(=O)(CC(CNCC)OC)N(CC(C)O)C.C(=O)CC(C)O 31156,N1(C(CN(CCC#C)C)=O)CCC2(COC(CNC(=O)CC3OCCCO3)C2)C1 31157,c1(CC(N2C(C(=O)OCC)C3C=CC2C3)C(=O)NC)cc2ccccc2o1 31158,N1(C(C2N(C)CCOC2)=O)CC2(CC(NC(C3(CC(F)F)CCNC3=O)=O)C2)C1 31159,N1(C(C(C)(C)CF)=O)CCC2(CC1)CCN(C(C1(n3cccn3)CCC1)=O)C2 31160,n1(CCCC)cc(C(=O)NC(C)(CNC(c2nc(C)oc2C)=O)CO)c(C)n1 31161,O=C(COCc1ccccc1)N1CCC(S(=O)(=O)Nc2ccccc2)C1 31162,C(=O)(C(C)(C)CC(=O)N1CCCC(N(C)C(C2CCCC2F)=O)CC1)OC 31163,C1(C(=O)NCc2n(C(C)C)ncn2)CCCCN(C(C2CC23CCC3)=O)C1 31164,N1(C(C2CCC2(F)F)=O)CCC(F)(CNC(C2(c3cccs3)CC2)=O)C1 31165,C(=O)(CC(C)CC(=O)N1CCOCC(C(=O)NCC(C)(C)OC)C1)OC 31166,N1(C(C(C)NC=O)=O)CC(NC(=O)C=CC2CCOCC2)CCC1C 31167,C1(NC(CNC(N)=O)=O)CCN(C(=O)CN2CCC2)C1 31168,C(CN=c1[nH]c(Cl)nc2ccccc12)NC(C(C(C)C)NC(C)=O)=O 31169,C(C(C(C)(C)C)NC(C1(C)COC(=O)N1)=O)NC(Cc1cn(C)nc1)=O 31170,c1(C(N(C)CC2CCC(NC(CC3C(OC)CC3)=O)CC2)=O)cc([N+](=O)[O-])c[nH]1 31171,C1(NC(CC)=O)(CO)CCCN(C(=O)C(COCc2ccccc2)N(C)C)C1 31172,c1(C(C)C)cncc(C(=O)NCC2CC(NC(=O)CCc3cccn3C)C2)c1 31173,c1(C(N(CC(CC)NC(c2cccnc2)=O)C)=O)c(C)oc(C)c1C 31174,N1(C(C2C(CC)C2)=O)CCC2(CCCN2C(=O)CSCc2cccnc2)C1 31175,c1(C(N(CC(C)O)CCNC(C2(C)CC=CC2)=O)=O)ccc(-c2cnn[nH]2)cc1 31176,C1(NC(CS(=O)(=O)NC)=O)CC2CC1CN(C(C1CC(C(F)(F)F)(OC)C1)=O)C2 31177,C(=O)(C(F)(F)C(F)(F)C(F)(F)C(F)F)NC1C(C)(C)C(C(=O)O)C1 31178,c1(-c2ncc(C(=O)NCC(CC)NC(=O)C(F)CC3CC3)s2)ccc(F)cc1F 31179,N1(C(CCc2c(C)ncs2)=O)CC2CC1C2NC(C1CC(C)(C)C1)=O 31180,C1(NC(C(C=C)(C)C)=O)CCN(C(=O)Cn2cncc2C(=O)OC)CC1C 31181,N1(C(CNC(CC)=O)=O)CC2CCC(C1)CC(NC(C13CCC(OC)C1C3)=O)C2 31182,c1(C(=O)NC(CC)CNC(=O)C(O)C2CCC2)c(NC(C)=O)cccc1F 31183,CC(CNC(=O)COC(F)(F)F)CNC(=O)C(F)C1CCCC1 31184,C1(NC(c2cc(-c3ccns3)on2)=O)COCCN(C(c2ccccc2)=O)C1 31185,N1(C(Cc2nc(C)[nH]n2)=O)CC(C(=O)Nc2ccc(F)nc2C)CC1(C)C 31186,c1(C(N2C(C)CC(CNC(=O)Cn3cnnn3)C2)=O)ccc2c(c1)nnn2C 31187,c1(C(=O)NC(CN(C(C2(COC)CC=CCC2)=O)C)C)ccc2ccccc2c1 31188,C1(NC(CCSCC)=O)CC2CCC1N(C(c1cc(C(N)=O)cs1)=O)C2 31189,O=C(C1=COCCO1)N1CCN(C(c2ccc(-c3ccco3)[nH]2)=O)C(CF)C1 31190,C1(CNC(C2(CCC)CC2)=O)CCC(NC(=O)Cc2nocc2C)C1 31191,Cc1nc(Cl)nc(N2CC3CN(C(C4CCS(=O)(=O)C4)=O)CC3C2)c1C#N 31192,C(C(C(=O)NCCC1(O)CCN(C(=O)C=CCO)C1)C(C)(C)C)OCC=C 31193,C1(NC(CCOCCOC)=O)CN(C(c2ccsc2)=O)CC1C 31194,CC(C)CC(C)(C)C(=O)NCC1CC(C)CN(C(=O)C(Cl)=CCl)C1 31195,C1(C(N(C)Cc2nnnn2C)=O)CC(=O)CN1C(=O)CSC1CC1 31196,C1(C(N2CC(CNC(c3c(C)nc[nH]3)=O)C(C)C2)=O)CCc2ncncc2C1 31197,C1(C2CC2)(C(=O)NCC(CC)(CC)NC(c2cnn(C)c2C)=O)CC=CC1 31198,N1(C(c2cc(OC)c(O)nc2)=O)CC2(CCN(C(c3nc(C)n(C)n3)=O)C2)C1 31199,CCCCCC(O)CC(=O)NC12CC1CN(C(=O)CC(N1CCCCC1=O)C)C2 31200,c1(CNC(C2(CC)CCOC2)=O)ncccc1C(N1CC(C)(OC)C1)=O 31201,N1(C(c2sc(C)c([N+](=O)[O-])c2)=O)CCC2(CCOC2=O)CC1 31202,C1(C(C)NC(=O)C(CN(C)C)N(C)C)CCCCN1C(c1ccc(C(F)F)s1)=O 31203,C1(C(N2CCCC2c2ccccc2)=O)(COC)CCCNC1 31204,C1(CC(N2CC(C)(CC(=O)OC)C2)=O)CC(N=c2cc(C)nc(C(=O)OC)[nH]2)C1 31205,C(N=c1[nH]c(=NCC2CCCCS2)[nH]c2c1COC2)c1c(Cl)c2c(s1)CCCC2 31206,C(CCCCC(=O)NCCC(O)C1CCCC1)N(C(C=CC(=O)OCC)=O)C 31207,CCCC(CNC(C1CCC(=O)N1C)=O)CCO 31208,c1(CC)c(C(=O)NCC(C)N(C)C(c2cccc(-n3ccnc3)c2)=O)nnn1C 31209,C(=O)(C(O)CC(F)(F)F)N(CCNC(c1c(Cl)n[nH]c1C1CC1)=O)CC 31210,c1(-c2scc(C(N(CCCNC(C(CC)SC)=O)CC)=O)n2)cccc(C#N)c1 31211,c1(CC)cnc(O)c(C(=O)NCC(C)(C)NC(c2cc(C3CC3)ccc2Cl)=O)c1 31212,C(CO)(CCCO)C(N1C(C(=O)NCCCCCF)CSC1)=O 31213,c1(C(N2CCC(CC=C)(NC(C3C4CCCC34)=O)C2)=O)ccc2c(c1)CCN2 31214,c1(CC)ccc(C(C)C(=O)N2CC(CCNC(c3cccnc3O)=O)C2)cc1 31215,C1(O)(C(C)NC(CC)=O)CCN(C(c2cccc(-n3cccn3)n2)=O)CC1 31216,C1(NC(CCCC#C)=O)CCCC12CCN(C(c1cc(N)nc(Br)c1)=O)C2 31217,c1(C(N2CC(OC)(CNC(=O)C(C)C(C)(F)F)C2)=O)cc(S(C)(=O)=O)co1 31218,N1(C(COCCCOC)=O)CCCN(C(=O)CN2CCC(C)CC2)CC1C(C)C 31219,CC1(C)C(CC(=O)NC(C2CCCCC2)C(=O)NCc2ccc(O)cc2)C1(C)C 31220,CC1CC(NC(C2CC3CCC(C2)S3)=O)CCN1C(c1cc2occc2[nH]1)=O 31221,N1(c2nnc(COC)s2)CCC2(CCC2)C(NC(=O)C2Cc3ccccc32)C1 31222,CC(C)C(C)C(CNC(C1(Br)CC1)=O)NC(C1(C(F)(F)F)CC1)=O 31223,C(=O)(C(=O)C(F)(F)F)N(CC(C)NC(C1(C)CCCO1)=O)C 31224,N1(C(CCC(=O)NCC)=O)CCCCC(C2CN(C(c3coc(Br)n3)=O)C2)C1 31225,N1(C(Cc2c(C)non2)=O)CCC(C2CCCCN2C(=O)COCCF)CC1 31226,Cc1cc(Br)cc(C)c1COC(=O)CCc1cccs1 31227,Cc1cc(CN2CCOC(C(N3CCC(CO)C(O)C3)=O)C2)c(C)cc1Br 31228,N1(C(c2cccn(C)c2=O)=O)CCCC(NC(=O)CCc2ccsc2)C(F)C1 31229,CCCCCCN(C(=O)CCC=C(C)C)CCCC.C1(=O)C(C)N1 31230,N1(C(CC=C)=O)CCOCC12COCCN(C(=O)CCCCC(C)CC)C2 31231,c1(C(N2CC(C)(c3cn(-c4ccc(Cl)nc4)nn3)C2)=O)nccc2cccnc12 31232,C(=O)(CCCCCNC(=O)CC1CC1(C)C)NC(c1nccs1)(C)C 31233,c1(C(C)C)ncc(C(=O)NCC23CC(CN2c2ccnc(C4CCC4)n2)C3)cn1 31234,c1(C(N(CCCOCCNC(C2CCS(=O)(=O)N2)=O)C)=O)cc(Cl)n[nH]c1=N 31235,c1(C(N2C(CC(N3CC(=C)C3)=O)COCC2)=O)cccc(C)c1C#N 31236,C(=O)(C1=C(C)CCOC1)NCCN(CC(C)O)C(c1cnc(CC)[nH]1)=O 31237,C1(C(=O)NC2CN(C(=O)C(=CC3CCCC3)C)C2)(OC)CCCOC1 31238,CS(=O)(=O)CC(=O)N1CCCC1CC1CCCN(C(c2ccc(Cl)cc2)=O)C1 31239,C(=O)(C1=CCC(F)(F)CC1)NCC1(C)CCC(NC(CC(CC)C)=O)CC1 31240,N1(C(c2c(C)scn2)=O)CC2C3CCC(C2C1)N(C(c1cccnc1O)=O)C3 31241,C(CCCC(=O)N1CC(OCC(=O)N(CCCC(O)CO)C)C1)N(C)C 31242,N1(C(COC2CN(C(C)=O)C2)=O)CCC2CN(C(=O)Cn3ccc(C)n3)CC12 31243,c1(C(=O)NC2CC2NC(C2(O)COC2)=O)cccc(Cn2ccnn2)c1 31244,c1(CC)cc(C(N2CCC2C(=O)N(C)C)=O)ns1 31245,c1(C(N2CCC3(CN(C(c4c(N)nccn4)=O)C3)C2)=O)cc2c(Cl)cncc2o1 31246,c1(OC)cc(N)c(F)cc1C(=O)NC1CC(C)(NC(c2cc(O)nc(Cl)c2)=O)C1 31247,C#Cc1ccc(C(N2CCC(NC(c3ccc(SC)o3)=O)C2)=O)cc1F 31248,C12CCN(C1)C(C1CC=CCC1)C(=O)NC21CC1.C1(C(N)=O)CC(F)(F)C1 31249,C1(NC(C2(CCNC(=O)C(F)n3ccnc3)CC2)=O)COCCC1(F)F 31250,c1(C(=O)NC2CCN(C(C3N(C(C)C)CCC3)=O)C(C)C2)nnc2n1CCCC2 31251,C12(NC(C3CCC4(CCC4)O3)=O)CCCC1N(C(c1cncs1)=O)CCC2 31252,N1(C(C(=O)N(CCNC(C(CC)(F)F)=O)C)CC)CCc2ccccc21 31253,CC1CC(C(=O)NCC2(C(=O)NCC(F)Cl)CC2)=NO1 31254,C1(NC(C2(C)CCCS2)=O)CC2(NC(c3cc(C(N)=O)co3)=O)COC1C2 31255,C(C)(CCCC(C)C)NC(C1C(CNC(C(COC)(C)OC)=O)C1(C)C)=O 31256,c1(OC)ccccc1C(CNC(=O)CCC1CC1C)NC(c1cc(=O)cc[nH]1)=O 31257,c1(C(=O)NC(C(=O)NC(C2(OC)CCC2)C)Cc2ccoc2)ccc(F)cn1 31258,c1(CCO)cccc(OCCNc2cc(I)ccn2)c1 31259,C1(NC(C2(CC)CC2)=O)CC=CCC1C(=O)N(CC(F)(F)Cl)C 31260,C1(NC(c2cc(Br)ccc2F)=O)CCCN(C(c2ccc(I)c(O)c2)=O)CC1 31261,c1(C2CC(NC3(c4nnnn4C(C)(C)C)CCN(C)C3)C2)ccc(F)c(Cl)c1 31262,N1(C(c2ncn(CC)c2)=O)CCC(C)C1CNC(=O)C=Cc1ncco1 31263,c1(C(=O)NC(CC(C)NC(c2cccc(C(C)=O)c2)=O)C)cc(C)c(C)nn1 31264,C1(C(=O)NCC2CCC3(CN(C(=O)CO)C3)O2)CCc2ccccc2O1 31265,c1(OCCCNCCCC(C)CC(=O)O)cccc(S(C)(=O)=O)c1 31266,CC(F)(C(=O)N1C2CCC1CN(C(c1ccc3cnnn3c1)=O)C2)C(F)(F)F 31267,C(C)(C(=O)N(Cc1cn(CC(C)O)nn1)CC1CC1)(C1CC1)OC 31268,N1(C(C=CCCC(C)NC(CN(C2CC2)CC)=O)=O)CCCCCC1 31269,C1(NC(c2c(C)cc(F)nc2)=O)CCC2CC1CN2c1nc(Cl)ncc1Cl 31270,C(=O)(C(CO)N(C)C)N(CC(=O)NC1(CC(=O)OCC)CC1)C(C)C 31271,C(CCCC(CO)NC(=O)COC(F)F)NC(Cc1cccc(OC)c1)=O 31272,C1(COC(C2C(C)C(=O)C2)=O)(CF)CCOCC1 31273,N1(C(C(CC)SC)=O)CC(=O)NCC1C(=O)NC(COC)C(=O)OC 31274,c1(C(=O)NC2CC(C(N3CCCC(OC)C3)=O)C2)ccc(Cl)c(C)c1F 31275,C1(C(=O)NC2(CC)CCCN(C(=O)C(C)=C3CCC3)C2)CC(C(C)=NO)C1(C)C 31276,N1(C(C)=O)CC2CCC(NC(c3ccnc(C(N)=O)c3)=O)(C2)C1 31277,c1(C(N2CC(CN(C(C3CCN(C)C3=O)=O)C)OCC2)=O)ccnc2ncnn12 31278,c1(C(=O)NCCN(C(CC(C)O)=O)CC(C)O)cnc2c(c1)NCC2 31279,c1(CC)nc(C)c(C(=O)NCCNC(c2nnsc2SC)=O)s1 31280,c1(C(N(C)CC2CC(F)CN2C(C2CCCO2)=O)=O)c(F)ccc(F)c1F 31281,C1(OC)CC2(C1)CC(NC(C1(C)CCN(C(C3CCC(=O)C(C)C3)=O)C1)=O)C2 31282,N1(C(COC)=O)C2CCCC1CN(C(=O)CCN1CCN(S(C)(=O)=O)CC1)C2 31283,c1(C(N2CC3(C(=O)NC4CCCC4(F)F)CC2CO3)=O)ccc2[nH]ccc2n1 31284,C12(C(N3CCCC(N(C(=O)C4=CSCS4)C)C3)=O)CC3CC(C(=O)N1)C2C3 31285,c1(C(N2CCN(c3nc[nH]n3)CC2)C(=O)NCC=C)cnc2c(c1)COC2 31286,c1(C(N2CCCC(C(=O)Nc3ccc(Cl)cc3CO)C2)=O)cc2ccoc2cn1 31287,c1(OCC)cnc(C(=O)NC2COCC2NC(=O)CCc2ccco2)c(Cl)c1 31288,CCC(COC)C(=O)N(CCNC(=O)C(c1ccc(Cl)cc1)C)C1CC1 31289,c1(SC)cc(C)c(C(=O)NC23CC2CN(C(=O)CC(C)NC(N)=O)C3)o1 31290,C1(C(=O)NC2CCC(CCC(=O)N(CC(F)(F)C(N)=O)C)C2)CC(O)C(F)C1 31291,C=CC1(c2ccccc2)COCCN1C(=O)C(=O)N1CC(Oc2ccc(Br)o2)C1 31292,N1(C(c2ccc(OCOC)cc2)=O)CC(NC(=O)CC2C(C)C2(F)F)CC(F)C1 31293,C1(C)(CNC(C2C(C)(C)C2)=O)CCN(C(c2cnn(C3CC3(F)F)c2)=O)C1 31294,c1(C(=O)NC2CCC(C)(NC(COC)=O)CC2)ccc2ncccc2c1F 31295,C1(NC(CN(C2CCSC2)C)=O)COc2cc(F)ccc2C1 31296,CCCC(=O)N(CCN(C(=O)Cn1cccc1)CC)CC 31297,C1(C(=O)NCC(C)(O)CN(C)C)(CC)CCNC1 31298,Cc1cc(NC(C2CCN2C(=O)Cc2ccc(Cl)s2)=O)cc(Br)c1 31299,Cc1ccc(F)c(C(N2CC3CC2CN3c2ncc(C3CC3)cn2)=O)c1Cl 31300,c1(CC)nc(C)cc(=NC(C)CC(C)NC(=O)C(C)(C)OC)[nH]1 31301,N1(C(CCC(=C)Cl)=O)CCN(C(=O)CC2CCC(F)(F)CC2)CC(O)C1 31302,N1(C(Cc2c(C)cccc2C)=O)CCN(C(c2cscn2)=O)CC(CO)C1 31303,c1(C(=O)NCC2CC(NC(COCC)=O)C2)ccccc1SC(C)C 31304,CCCCCCCC(F)C(=O)N1CCOCC12CCCC2 31305,C(=O)(CCN=C(NCC(C1CCCCO1)(C)C)NC1CC=CC1)N(C)C 31306,CC1(C)CN(C(C2(CNC(c3cc(CO)ccn3)=O)CCC2)=O)CCC1CO 31307,Cc1scc(C(=O)NCC(C)(O)CNC(c2cccn2C2CCCC2)=O)c1N 31308,C(=O)(C(CC(C)C)CNCc1ccccc1OC(C)C)OCC 31309,C(=O)(C(C)(O)C(C)C)N(CCCN(C)C)CCNC(c1ncc(OC)nc1)=O 31310,Cc1occ(C(F)(F)F)c1C(=O)NCCC1(O)CCN(C(C2(CF)CCC2)=O)C1 31311,c1(C(=O)NC(C2CCOC2)C)ccc(CNC(c2coc(N(C)C)n2)=O)cc1 31312,C1(C(=O)NC2CCN(C(=O)CCc3ncc[nH]3)C2C2CC2)CCCS(=O)(=O)C1 31313,C1(NC(c2n(CC)cc(Cl)c2)=O)CC2CN(C(C3(O)CCC3)=O)CC2C1 31314,CCC(C)(C(=O)N(C)CC1(CNC(C2CCCC(C)(C)C2)=O)CC1)C(N)=O 31315,C1(NC(C(CNC(=O)COC2CC=CC2)N(C)C)=O)CC2CCC1O2 31316,c1(C(N(C(C(=O)N(CC(C)OC)CC)C2CC2)C)=O)ccc2c[nH]nc2c1 31317,Cc1ccc(N)cc1C(N1CCCC(CO)(NC(=O)Cn2nnnc2C)C1)=O 31318,N1(C(C2CC(Cc3cn(COC)nn3)C2)=O)C2CCCC1C(C(=O)O)C2C(C)=O 31319,CCC(C(=O)N1CCC(NC(=O)CN2CCN(C)C(=O)C2)C1C(C)C)C(F)(F)F 31320,c1(C(=O)NC(CC(CC)C)C(=O)NCCOC)noc2ccc(Br)cc12 31321,C1(N(CCNC(CCCC)=O)C(c2csc(-c3ncc[nH]3)n2)=O)CCCCCC1 31322,C(C)(C(=O)N1CC(C(O)C(=O)NCCn2ccnn2)C1)OCCCC 31323,C(=O)(C(O)CC(N)=O)N1CCC(C(=O)Nc2cn(CC#C)nc2)(OC)C1 31324,N#Cc1c[nH]c(C(N2CCC(C(N3CCN(c4ccccc4)CC3)=O)CC2)=O)c1 31325,C1(NC(CC2(C=C)CCC2)=O)CCCN(C(c2cccnc2C(F)F)=O)CC1F 31326,N1(C(C(c2cnn(C)c2)NC)=O)CCc2ncc(CO)cc2C1 31327,c1(C(=O)NC2C3CC(OCC)C(C3)C2)noc2c1CC(F)(F)CC2 31328,CCCC(O)C(=O)NCC12CC(CN1C(=O)CC(C)N(C)C(=O)OC(C)(C)C)C2 31329,C1(C(C)(C)C)(CNC(CC(C)c2ccco2)=O)CCN(C(c2cccnn2)=O)C1 31330,c1(NC(=O)CCC2CCCN2c2ccn3nccc3c2)cc(Br)c(O)cc1Br 31331,CCC(CCC(=O)N1CCC(C)C1NC(=O)C=CC(=O)NC1CC1)OC 31332,C1(OC)CCCCC1N=c1cc(C)[nH]c(=NCCN(C)Cc2ccccc2)[nH]1 31333,N1(C(c2c(C)cco2)=O)CCC(C2CCN(C(=O)CC3COC(C)(C)C3)C2)CC1 31334,C1(C(=O)NC(C)C(N)=O)C2CCC1CN(C(c1cc3ccoc3cn1)=O)C2 31335,c1(OCC(=O)NC2C(NC(c3c(C)cno3)=O)C2)cccc(Br)c1C#N 31336,C(C(C)(O)C(=O)N1CC(NC(=O)CCc2c(C)noc2C)C(C)C1)OC 31337,c1(CCC)c(C(=O)N(C2CCCN(C(=O)C(F)=C(C)C)C2)C)nnn1CC 31338,c1(C(N2CCC(C)(c3cn(Cc4ncon4)nn3)C2)=O)nc(Cl)ncc1OC.CO 31339,CC1(c2cn(-c3ccc(C(=O)O)cc3)nn2)CCCN1C(C1CCOCC1)=O 31340,Cc1ccc2c(C(=O)NC3CCC4CCN(C(c5cccs5)=O)C3C4)n[nH]c2c1 31341,N1(C(C(C)C)=O)CCCCC1C(C)NC(=O)CCCc1nccs1 31342,C(=O)(C(CC)CC(F)F)N(CC(CNC(CCOCCOCC)=O)(C)C)C 31343,N1(C(c2nc(=N)[nH]cc2)=O)CC(F)(F)CC1C(=O)NC1C(O)C2CCOC12 31344,C1(C(CNC(C2C(OCC)C2)=O)(C)C)CCCN1C(=O)C(=O)Nc1ccccc1 31345,C1(C)(C(=O)NCC(C2CCCCC2)NC(Cc2c(C)con2)=O)CCCCO1 31346,N1(C(CCCC#C)=O)CCC(NC(=O)C=Cc2ccc(C(N)=O)cc2)CC1C 31347,C1(CC)(NC(=O)CSCC(C)C)CCCN(C(c2ccnn2CC(F)(F)F)=O)C1 31348,CC1(C)CN(C(=O)Cc2ccccc2Br)CC1NC(C1C2CCCC12)=O 31349,c1(NC(CCCC=C)C)ncc(S(=O)(=O)NCC2CCCCN2CC)cc1Cl 31350,c1(CC(C)NC(c2c(C)nc(CCOC)s2)=O)cc(F)c(F)cc1Br 31351,C(=O)(C#CC1(C)CCCO1)NC1CCC(NC(c2cc(C)cc(Cl)c2N)=O)CC1 31352,C1(COCC(=O)OCC)CN(N2CCCCC2C)C1 31353,Cc1cc2ccccc2nc1C(=O)OC(C)C(c1ccc(F)c(N(C)C)c1)=O 31354,C1(NC(CCC=C(C)C)=O)CC(C)CN(C(=O)Cc2ccc(C3CCC3)cc2)C1 31355,C(=O)(C1=NOC2(CCC2)C1)NC1C(NC(=O)CCC(=O)c2cccnc2)CCC1 31356,N1(CC)CCCCC(N=c2[nH]c(=NC3CC(CO)C3)[nH]c3c(F)cc(F)cc23)C1 31357,C(=O)(C1=CCS(=O)(=O)C1)N1CCC(NC(C(C(=C)Cl)(C)C)=O)C(F)C1 31358,C(C)(CSC)(C(=O)NCCCC(F)(F)F)NC(c1cn(CCC)nc1)=O 31359,N1(CC(=O)OCCCCCF)CCN(C(c2cnco2)=O)CC1 31360,C1(C#N)(C(=O)NCC(CC)(CC)NC(=O)CC2CCC(=O)N2)CC12CCC2 31361,N1(C(CC(C)(C)CO)=O)CCN(C(C2C3CN(CC(F)(F)F)CC23)=O)C(C2CC2)C1 31362,C1(CC)CN(C(=O)CCNS(=O)(=O)C(F)F)CCC1NC(C1(CCOC)CC1)=O 31363,N1(C(CCCCCC)=O)CC2CC3CC2C1C3NCC(=O)OC(C1CCCC1)=O 31364,c1(C(C)=O)c[nH]c(C(N2CCC(O)(C(C)CNC(c3csc(F)c3)=O)C2)=O)c1C 31365,CC1(C)COC(CC(=O)NC(C(=O)N2CC(C(C)(C)C)C2)c2cccs2)C1 31366,C1(CCCNC(C2C(C(=O)OC)C2)=O)CCCN1C(C1CCC(=O)C1)=O 31367,C1(C(=O)NC(CSCC)CO)C2CC3C(C2NC(C2(C)C(C)(C)C2(C)C)=O)C13 31368,N1(C(c2scc(C)c2)=O)CC(CNC(C2SC3C=CC2CC3)=O)C(C)(C)C1 31369,n1(CC)nc(C(=O)NC2CC23CC(NC(=O)C(C)NC(N)=O)C3)c(C)n1 31370,C1(NC(=O)NCC2(F)CCOCC2)COC2(CCOCC2)C1 31371,c1(CCC)ncc(NC(=O)C(C)(C)CN(C(=O)C=CC2CCOC2)C)cn1 31372,c1(CC)nc(C(N2CC(CO)(NC(c3scnc3C(C)C)=O)C2)=O)cs1 31373,C#Cc1ccc(C(N2CC3CC(NC(C45CCCC4CCC5)=O)C3C2)=O)nc1 31374,n1(CC(=O)NCCOCCN(C)C(C2(n3cnnn3)CC2)=O)cnc(=N)[nH]1 31375,N1(C(C(C)NC(CC)=O)=O)CC(F)(F)CC1CNC(c1cccc(C)n1)=O 31376,c1(-c2cc(C)no2)cccc(CNC23CC(C(=O)NC(C#N)C(N)=O)(C2)C3)c1 31377,S(=O)(=O)(c1ccc(Br)cc1NCC1OCCCO1)N1CCCC(CS(N)(=O)=O)C1 31378,c1(SCC)nccnc1C(=O)NCC(C(C)C)NC(C1(CC)CCC1)=O 31379,CC1C(NC(C2CCC2)=O)CC2CCC1N2C(=O)CC1CC(F)(F)C1 31380,C1(C(=O)NCCCCNC(c2c(C)n(C3CCOC3)nn2)=O)CCCS(=O)(=O)C1 31381,c1(C(C)NC(c2ccnnc2)c2nnnn2CCF)cccnc1 31382,c1(C(=O)NCC2(F)CCC(NC(C3CCS(=O)(=O)N3)=O)C2)ccc2nn[nH]c2c1 31383,Cc1ccncc1CC(=O)NC1CN(C(=O)Cc2ncc(Cl)s2)CC1C 31384,c1(C(N2CCC(CNC(C(C)SC)=O)C23CCC3)=O)ccc2ncc(=O)[nH]c2c1 31385,C1(c2cn(CCN(C)C(c3cncc(OCC(F)(F)F)c3)=O)nn2)COCC1(C)C 31386,C1(CCNC(C2CCN(C(CC)=O)C2)=O)CCCN(C(c2n[nH]cc2CC)=O)C1 31387,C(N=C(NC1CC1C)N1CCn2c(n[nH]c(=O)c2=O)C1)c1c(OC)cc(C)cc1 31388,C(=O)(CCC(C)NC(=O)Nc1ccc(C2(C)CC(=O)C2)cc1)OC 31389,CCCCC(C(=O)N1CC(C)(C#N)C1)NC(=O)CC=CC(C)(C)C 31390,c1(C(N(C(CCNC(c2c(C)cc(C)s2)=O)C)C)=O)ccc(S(=O)(=O)CF)nc1 31391,C1(CNC(C(C)OCCC#C)=O)CC2CN(C(C3(CC)CCCCC3)=O)CC12 31392,c1(C(N2C(C(N(C)CC3CCCO3)=O)COCC2)=O)ccc(O)c(F)c1 31393,CC1SCCC1NC(C1(CCNC(C2CC3(CC3)C2)=O)CCCC1)=O 31394,c1(OC)ccccc1C(CNC(=O)Cc1[nH]cnc1C)NC(=O)C(C)C(C)C 31395,C1(O)(CC#C)CCN(C(c2ccc(COC(C)=O)cc2)=O)CC1 31396,C1(F)(CNC(C(F)=C(C)C)=O)CCCN(C(=O)CCCC2CCC2)CC1 31397,CCC1=NOC(C(=O)NCCN(C(=O)CCc2ccncc2Br)C)C1 31398,C(C)(CCC(=O)NC(Cc1cc[nH]n1)C(=O)NCCc1nccs1)OC 31399,C1(C(CNC(CC(C)F)=O)(C)C)CCN(C(c2cnn(C)c2C(F)(F)F)=O)CC1 31400,C1(CNC(CCSCCC)=O)CCCCN(C(C2(C)CSC2)=O)C1 31401,C(CC(=O)NC(C)CSc1cnc[nH]1)N(C(C)C)C(C1CN(C2CCC2)C1)=O 31402,N1(C(c2cncc(CC)c2)=O)CC(NC(=O)C(C)NC(=O)C2CC2)CC(O)C1 31403,N1(C(C2C(C)(C)CC(=O)NC2)=O)CC23CCCC2(C1)CN(c1ncc(F)cn1)C3 31404,N1(C(c2c(C)ncc(N)c2)=O)CC2CCCC(C1)N2C(=O)C(C)(O)C1CCOC1 31405,C(=O)(C1=C(C)C(C)(C)OC1=O)NC1CCCCN(C(C(CNC(C)=O)(C)C)=O)C1 31406,Cc1cc(C)c(C#N)c(NC(C2CCCN(C(c3ccc(Cl)nc3)=O)C2)C)n1 31407,c1(OC)ccc(C=CC(=O)NC2CCN(C(C3(C)CC3(F)F)=O)CC2O)cc1Cl 31408,c1(C(=O)NC2C(NC(C3(OC)CCC3)=O)COC2)sc([N+](=O)[O-])cc1Cl 31409,c1(C(=O)OC)cc(C(=O)NC2CN(C(=O)CSCCC(C)C)CC2C)n(C)n1 31410,c1(OC)cnc(F)cc1C(=O)NC1COCC1NC(=O)C=CC1CCCC1 31411,C(=O)(C(C)CC(=O)OC)N1CCC(N2CCC(NC(CNC(CC)=O)=O)C2)CC1 31412,N1(C(C2CCC(C)(CC)O2)=O)CCC2CCN(C(=O)C(CC)(CC)OC)CC12 31413,c1(C(N2CCN(C(C)CNC(C3(CC4CC4)CC3)=O)CC2)=O)nccn2nccc12 31414,c1(C(N2C3CN(C(C4(O)CC(C)(C)C4)=O)C(C3)C2)=O)cc2n(n1)CCC2 31415,C1(CN(CC(=O)NC(c2cnn[nH]2)C)C2CC2)CCN(C(C2CC2)=O)CC1 31416,c1(C(N2CC(C(N(CC(C)O)CC(C)O)=O)C3(C2)CC3)=O)nccc2cc[nH]c12 31417,c1(CC(=O)NCCC2(O)CN(C(=O)C=Cc3cnc[nH]3)C2)sccc1Br 31418,c1(C(=O)Nc2cccc(-c3ccc(O)cc3)c2)cc2cncn2c(O)n1 31419,N1(C(c2c(NC)nccc2)=O)CC2(CCCCN2C(C2(CF)CC2)=O)C1 31420,C12(NC(COC)=O)CC(CNC(C3(Cl)CC3(F)F)=O)(C1)OC21CCC1 31421,C1(NC(C(C2(NC(c3cc(SC)oc3)=O)CCC2)O)=O)CCCCC1CO 31422,c1(OC)c(C(N2CCC(CNC(C3CC3C(=O)NCCO)=O)C2)=O)ccnc1Cl 31423,C1(C(=O)NCC(CC)NC(=O)CC2CCCO2)(OC)CCS(=O)(=O)C1 31424,N1(C(=O)NC(C2CCC3(CC3)N2C(=O)OC(C)(C)C)C)CCCc2ccccc21 31425,c1(C(N2CCC(N3CCN(C(C)=O)CC3)C2)=O)ccc2c(n1)OCCO2 31426,c1(C(=O)OC)nn(C)c(NC(C2CN(C(C3CN(C)C3)=O)CCS2)=O)c1Cl 31427,CCCCN=C(NCCC1(NC(=O)OC(C)(C)C)COC1)NC1CCS(=O)(=O)C1 31428,N1(C(CCc2ccn(C)c2)=O)CCC2C(C1)CN2C(C1CCCNS1(=O)=O)=O 31429,C1(NC(c2cnsc2)=O)CCOC2(CCN(C(c3ccncc3O)=O)CC2)C1 31430,Fc1cc2nc(-n3nc(C4CCOC4)nc3CC3=CCOCC3)[nH]c2cc1F 31431,C1(C(=O)NCC(C)(C(C)C)NC(c2c(OC)n(C)nc2)=O)CCN(C)C(=O)C1 31432,N1(C(C2(C)CCSCC2)=O)CCC(F)C(NC(C2(CC3CC3)CCOCC2)=O)C1 31433,C(=O)(C(C)CC(C)C)N1C(C2CCN(Cc3nc(CC)on3)C2)CCC1 31434,N1(C(c2ccc(NC)c(F)c2)=O)CCC2CCN(C(C3CC=CC3)=O)CC12 31435,c1(C(N2C(C(N3CCC(CN(C)CC)C3)=O)C=CC2)=O)ncccc1Cl 31436,N1(C(=O)NC)CCC(C(=O)NCC#CCNC(c2sccc2-n2cnnn2)=O)C1 31437,CCC(CCOC)C(=O)N1CC2CC(C1)C2NC(=O)CC1C(=O)NN=C1C 31438,c1(NC(C)=O)cccnc1C(N1CCOC(C(C)NC(=O)CCNC(N)=O)C1)=O 31439,C(=O)(CC1=CCN(C)CC1)NC(CCC)C(O)C(=O)NCCCC1CCOC1=O 31440,C1(CN(C(=O)Nc2cnco2)CC)CCCN(C(=O)OC(C)(C)C)C1 31441,Cc1nc(C)c(C(=O)NCC2CCOC2C(=O)Nc2ccc(C(C)C)nc2)s1 31442,CC(CC1CCCO1)C(=O)N(CCCOCCNC(c1csc(O)n1)=O)C 31443,C1(CNC(C2CCC(C)(C)C2)C)CCCC(F)(F)C(=O)N1 31444,C1(C(N(CC=CC(=O)N(C(C#C)C)C)C)=O)CC(OC)(OC)C1 31445,C1(CC)CCN(C(c2cc(C)oc2C)=O)C1CNC(=O)C=CC1CCOC1 31446,C(=O)(C(C)(C)C(F)F)NC1CCC(F)(CNC(c2ccc(CC(C)C)s2)=O)C1 31447,C1(C(=O)NCCCCN=[N+]=[N-])CCN(C(C2(CO)CCCCC2)=O)CC1O 31448,c1(CNC(=O)NCCNC(CC)=O)ccc2c(c1)CCCCN2 31449,O=C(CCC(F)(F)F)NCC12CC1CN(C(c1cncc(O)c1)=O)C2 31450,CCC(CNC(C1CCOC(C)C1)=O)(CC)NC(c1ccnnc1S)=O 31451,C1(C(C)C)(C(N2CCC(C(C)NC(=O)Cc3ccc(Cl)s3)CC2)=O)CNC(=O)C1 31452,CN1CC(F)CC1C(N1CC(OCCNC(C2CC2[N+](=O)[O-])=O)C1)=O 31453,C1(COC)(CNC(C2C(C)C2C)=O)CCN(C(=O)Cc2cnc(C)[nH]2)CC1 31454,C1(CNC(C(CC)(C)COC)=O)CC2CCC(C1)N2C(=O)C1=NOC(C)(C)C1 31455,C1(O)(CNC(c2occc2C2CC2)=O)CCCN(C(C2CCCO2)=O)C1 31456,C1(C(=O)NC(CC)CNC(C2C3(CC3)C23CC3)=O)CCc2c(ncn2C)C1 31457,C1(NC(c2cn(CCC)nn2)=O)CC2CC1N(C(c1nnc(O)nc1O)=O)C2 31458,N1(Cc2ccc(OC)nc2OC)Cc2[nH][nH]c(=NC(=O)c3sccc3F)c2C1 31459,c1(C(N2CCN(CCCNC(CCC(C)OC)=O)CC2)=O)cc2c(ncn2C)[nH]1 31460,Cc1c(C(=O)NC2CN(C(C3CCC4(CC4)C3)=O)C(C)(C)C2)cccc1C#N 31461,C1(CNC(=O)NC(c2n[nH]c(C3CC3)n2)C)CC(C(F)(F)F)CO1 31462,C1(C(=O)NCC2CCCC2CF)(CC)CN(C(=O)COc2ccsc2)C1 31463,Cc1sc(Cl)nc1C(=O)NC1CN(C(c2ccccc2Br)=O)C2CC12 31464,C#Cc1ccccc1CC(N1CCOCC1CNC(C1CN2CCC1CC2)=O)=O 31465,N1(C(C(CCC)NC(CC(C=C)CCC)=O)=O)CCC2(CCC(OC)C2)C1 31466,c12cccc(c1)C(=O)N2.C1(CNC(c2cn(CC)cn2)=O)CCCN1CC 31467,C(C1CN(C(c2cc[nH]c2)=O)CC1C(=O)Nc1cnc(CO)nc1C)=CC 31468,c1(COC(C)=O)ccc(C(=O)NC(C)(C)CCCNC(=O)CC2CCOCC2)cc1 31469,C(=O)(N=c1cc(-c2cncc(Br)c2)o[nH]1)N(CCN1CCCC1=O)CC 31470,c1(C(C)C)ccc(N)c(C(N2CCN(C(=O)C3=CCC3)C(CO)C2)=O)c1 31471,N1(C(c2c(C)cns2)=O)CC(C(=O)NCCn2nncc2C)CCC1C 31472,CC1CCN(C(c2sccc2F)=O)CC1NC(c1cc(F)c[nH]1)=O 31473,Cc1cc(C(=O)NC2CC(NC(C3CCC(C(N)=O)O3)=O)C2)cc(N)c1O 31474,C(CC(CC)C(=O)N1CCCC1C(C)(C)NC(=O)CCCC1CCOCC1)=CC 31475,C12(N(C(CSc3n[nH]c(=N)s3)=O)CC3CC3)CCC(CN(C(=O)C3=COCC3)C1)C2 31476,c1(C(=O)OC)ccccc1C(=O)N(CC(C)N(C(=O)C(C)Cc1ccco1)C)C 31477,N1(C(C(CC#C)NC(C)=O)=O)CC(C2CN(C(c3ccc(N)c(OC)c3)=O)C2)C1 31478,C1(C(N2CC(NC(=O)CC3(O)CCC3)C2)=O)C2C3CCC(C3)C12 31479,C(=O)(CCCC(C)C)NCC1(CNC(c2c(SCC)cccc2)=O)CC1(F)F 31480,C(=O)(C(F)CC(C)C)N(C(CCNC(C1(CC=C)COC1)=O)C)C 31481,CC(O)C(O)CNC(=O)CCC1CCC(NC(C2CCO2)=O)C1 31482,c1(NC(N2CCCC(NC)C2)=O)cccc2c1ccn2CC(=O)NC 31483,C1(C)(CC)C=C(C(=O)NCC(C)N(C)C(c2ncc(Br)cc2C)=O)C1 31484,C(=O)(C=CS(C)=O)NCC1C(NC(C=CC=CC)=O)COC1 31485,C1(C)(C(N2CC(CNC(c3ccc(C(C)=O)nc3)=O)C(O)C2)=O)CCCS1(=O)=O 31486,N12CCC3(CC1)CC(C3)NC(=O)CCS2(=O)=O.c1(C(=O)OC)cc2sccc2s1 31487,C(=O)(C1Cc2ccccc21)NC12CCC(CN(C(c3c(C)cnnc3)=O)C1)C2 31488,c1(C2(NC(=O)NCC(C(C)O)O)COC2)ccc(Cl)nc1O 31489,C(=O)(CS(=O)(=O)CCOC)NCCCN(C(c1cc(CO)on1)=O)CC 31490,CC(C)CCCC(=O)NCCC1CCN(C(c2cnn(C)c2)=O)CC1 31491,N1(C(=O)OC(C)(C)C)CCC(CC(=O)OCc2c[nH]nc2-c2cnn(C)c2)C1 31492,CC(C)C(C)(CNC(c1ncoc1C1CC1)=O)NC(=O)CN1CC2CCC1C2 31493,c1(CN2C(CNC(c3c(C)cc[nH]3)=O)CCC2)ccc(C(F)(F)F)cc1Br 31494,c1(C(=O)NCC2CCCN(C(C3C(C)(CC)C3)=O)C2)noc2cc(Cl)ccc12 31495,c1(C(N(CC(C)NC(=O)C(O)CN(C)C)CC)=O)cccc(NC(C)=O)c1 31496,C(C(C(=O)NC1(CC)CCN(C(=O)C(CCC)CC)CC1)C(C)(C)C)OCC=C 31497,C(=O)(CCCC(N)=O)NC(C1CCN(C(c2ncccc2O)=O)CC1)C(C)C 31498,CC(CCC(C)(C)C)C(=O)NC1(CF)CCN(C(=O)C(C)(C)CF)C1 31499,c1(N(C2CC3(CNC3)C2)C(=O)Cc2cc(O)nnc2O)cc(F)c(F)cc1Br 31500,c1(C(N2CCC(C)(NC(=O)Cc3nnc(O)s3)C2)=O)ccc(Cl)c2cccnc12 31501,CC(CCCNC(c1cc(Cl)c[nH]1)=O)NC(=O)COCC(c1ccccc1)C 31502,Cn1nc(C(F)F)cc1S(=O)(=O)NCCc1cccc(Cl)c1 31503,C(C(=O)NCC(F)=C(C)C)(C1CCOC1)NC(C1(OCC)CC1)=O 31504,C1(C(=O)NCCN2CCOCC2)(CNC(CN(C2CCSC2)C)=O)CCCC1 31505,C(=O)(CCC(F)(F)F)N1CC(OCC(=O)NC2CCC2)C(C(F)F)C1 31506,C(=O)(C(C)(C)C(C)(C)O)NC1C=CC(CNC(C(C)c2cc[nH]n2)=O)C1 31507,Cc1nc2ccccc2cc1SC1CC2(CC(C(=O)O)C2)C1 31508,c1(SC)nc(N2CC3CCC2C(NC(=O)Cn2ncn(C)c2=O)C3)c(C)c(Cl)n1 31509,O=C1CCC(NC(c2conc2CNC(=O)CCCN2CCCC2)=O)C(=O)N1 31510,C(=O)(CC1OCCc2ccsc21)N1CC(NC(CC2C(C)(C)C2(C)C)=O)C1 31511,C1(NC(=O)NCC2(C)COC2)CCOC2(CCOC2)C1 31512,C1(C(=O)NCC2(CC)CCCC2)CCN(C(=O)C(C)n2cccn2)C(C)(C)C1 31513,c1(CN(C2C3CNC2C3)CC(=O)OCCCC)ccc(OC)cc1 31514,Cc1[nH]nc(C(N2CC3C(NC(=O)C(C)(C)n4cc(Cl)cn4)C3C2)=O)c1F 31515,C1(COC)(CNC(c2ccc(C(N)=O)o2)=O)CCN(C(=O)C=C(C)C)C1 31516,c1(CC)ncc(CNC(C2(CCNC(=O)C=CC3CC3)CC2)=O)[nH]1 31517,c1(OCC(=O)NCC(CC)(CC)NC(CCC#CC)=O)ccc(C(C)C)c(C)c1 31518,C#Cc1ccc(C(=O)NCC2(C)CCC(NC(c3cc(OC)nn3C)=O)C2)cc1 31519,c1(C(=O)NCC2CC2NC(C2CCC3(CC3)C2)=O)cc(=O)c2ccncc2o1 31520,c1(OC)ncc(C(N2CCCC2C(c2ccccn2)=O)=O)c(C)c1Br 31521,CC1(C)CN(C(c2cccc3ccoc23)C(=O)NC2CCC2)c2cccc(Cl)c21 31522,N1(C(c2cc(C3(C)CC3)n[nH]2)=O)CCCCC1CN(C(C1CCOC1=O)=O)C1CC1 31523,c1(CC)nnsc1C(=O)NCC1(C(N2CC(SC(F)F)C2)=O)CCCO1 31524,N1(C(C2(CSC)CC2)=O)CC(C2(NC(c3cnc(S)n3C)=O)CC2)C1 31525,Cc1cccn2cc(C(=O)NCC3C(O)C(O)CN3C(C3(F)CCOC3)=O)nc12 31526,c1(CN2CCCC(NC(c3ccnc(OC)c3F)=O)CC2)ccc(C#N)cc1F 31527,N1(C(c2c(-c3c(OCC)cc(F)cc3)c[nH]n2)=O)CCC2(CC1)OCCO2 31528,Cc1nc(C#N)c(NCCC(N2CCN(C(=O)C(C)(C)C(N)=O)C3CC23)=O)o1 31529,C1(C(N2CCC(C(C)(C)NC(C(C)=CC)=O)C2)=O)CCc2[nH]nc(O)c2C1 31530,N#CC1CCCC(C(=O)NC(Cc2ccco2)C(N2CC(F)CC2CO)=O)C1 31531,c1(C(=O)NC2CC(CNC(C(CC=C)C)=O)C2)ccc(Cl)cc1-c1ccccc1 31532,Cc1ccc(C(=O)N(C)CCN(C(=O)C(C)OCCN(C)C)C)c(Cl)c1 31533,C1(OC)CCC(C(=O)NCCC2(NC(=O)Cc3csc(C(C)OC)n3)CCC2)C1 31534,O=C1OC2CC(C(=O)NCC3CCCN3C(c3cnc4[nH]ncc4c3)=O)CC2O1 31535,C(C)(CCCCNC(c1ccc(F)cn1)=O)NC(C(N1CCSCC1)C)=O 31536,Cc1ccnnc1C(N1CC(CNC(=O)CNC(C2CCOCC2)=O)C(C)C1)=O 31537,c1(COC)nc(NC2CNC(=O)C2)cc(=NC2CC3COCC(C3)C2)[nH]1 31538,N1(C(CC2C(=O)NC(=N)S2)=O)CC(NC(C2CCC3(CCC3)C2)=O)CC(O)C1 31539,c1(OC)cccc(C(=O)NC2CCCCC2NC(=O)CNC(c2cscn2)=O)c1 31540,CCC(C(=O)NCC(O)CCNC(=O)Cc1csc(C(C)C)n1)NC(C)=O 31541,n1(CC)nc(C(N2CCOC(CNC(=O)C(C)CCOC)C2)=O)cc1C(F)(F)F 31542,C12(NC(c3ccc(C)c(F)c3)=O)CCOCC1CN(C(=O)C1CC1)C2 31543,C(=O)(C#CC(C)(C)C)NCC(C(=O)NC1CC2CC(O)C1C2)N(C)C 31544,c1(C(N(CC(=O)NC(C)CN=[N+]=[N-])C)=O)ccncc1F 31545,Cc1ccc(F)c(C(N2CC(NC(c3c(C)nc(C)nc3C)=O)C(C)C2)=O)c1Cl 31546,c1(C(N2C(C(=O)Nc3ccc(Cl)c(O)c3)CC2)=O)cnc2c(Br)cccc2c1 31547,c1(C(N2CCC(CNC(C(CCC#C)O)=O)C2(C)C)=O)ccc2occc2c1 31548,n1(CCOCC)cc(C(N2CC(NC(c3cc(C4CC4)cs3)=O)C2)=O)nn1 31549,c1(OC)ccc(C)c(N2CCCC2=O)c1.c1(NC)nnc2n1C2.C1(O)CCOC1 31550,c1(C(N(C2CCN(C(c3cncn3C)=O)C2)CC)=O)c2c(nn1C)CCCC2 31551,c1(CN2C(C(N(CCCN(C)C)CCC)=O)CCC2)cc(C(F)(F)F)ccc1C 31552,C=CC(C)(C)CCNC(=O)C(CNC(c1ccnc(CC)c1)=O)N(C)C 31553,C1(CC(=O)NC(C2(O)CCCCC2)C(=O)N(C2CC(F)(F)C2)C)CC2CCC1C2 31554,n1(CC(=O)NC23C(CN(C(C45CC(OC)C4C5)=O)C2)C3)nc(O)c2c1CCCC2 31555,c1(CNC(CCN(C(=O)Cc2ccsc2)C)=O)cncc(F)c1 31556,CCC(C)CC(=O)C(=O)N1CC(C(=O)NCCCCCCF)C(F)C1 31557,c1(NCC(C)(C)C2(O)CNC2)ncc(N2CCCCC2)cn1 31558,c1(C(=O)OC)ccc(-c2nc(Br)ccc2C)cc1C 31559,c1(CC)c(C(=O)N(CC(C)NC(=O)C(c2ccc(Cl)s2)=O)C)cnn1CC 31560,N1(C(C2N(C(C(C)OC(C)=O)=O)CCN(C)C2)=O)CC(C)OC2(CCC2)C1 31561,c1(C(=O)NCC2(C(=O)NC(CCOC)C)CCCO2)cccc2c[nH]nc12 31562,Cc1cccc(CCC(N2CCN(C(=O)C(O)C(C)(C)C)C(C)C2)=O)c1Br 31563,C=C(C)CCC(=O)NCc1nc(C2CCN(C(C3CCCN(C)C3)=O)CC2)n[nH]1 31564,C(N=c1[nH]c(=NCc2ccc(F)cc2)[nH]c2cc[nH]c12)c1cc(CC)[nH]n1 31565,CC1CN(C(C2CC(n3ccnc3)C2)=O)CCC1NC(c1ccc(O)nc1)=O 31566,C(=O)(C(C(C)C)N1CCCCC1)NCC1C(NC(C2CC(C)(CC)C2)=O)COC1 31567,N1(C(CCCCSC)=O)CC2CCCN(C(=O)CCc3cc(C)[nH]n3)C2C1 31568,C=CCCCCCCCCC(=O)N(C)CCNC(C1CC2OC(=O)OC2C1)=O 31569,c1(C(=O)NCC2N(C(c3cncc(CC)c3)=O)CCOC2)cc(Cl)c(F)cc1F 31570,C1(C(=O)NC2(COC)CCN(C(=O)Cc3ccco3)C2)(COC)CCC(=O)N1 31571,C(N=c1[nH]c2cc(F)ccc2o1)C1CCN(C(c2cccc(OCC)c2)=O)C1 31572,Cc1cc2[nH]c(C(N3CCC(C)(NC(C4CCC5(CCC5)C4)=O)C3)=O)cc2s1 31573,C1(C(N2CCC(c3cn(-c4cn(C)nc4C)nn3)C2)=O)(OC)CCS(=O)(=O)C1 31574,N1(C(C(C)OCC)=O)CCC2CN(C(c3cc(OC)nc(OC)c3)=O)CC2CC1 31575,C(=O)(C(F)(CNC(=O)Cn1ccnc1)C(C)C)NC(C#C)C(C)OC 31576,CC(CN=c1[nH]c2cccc(F)c2s1)(C1CC1)NC(c1cc(Cl)cs1)=O 31577,Cc1nn(C)c(NC(=O)C(C)Cc2cnc[nH]2)c1Br 31578,N1(C(C)C)CC(NC(=O)CC2CN(C(c3cc(CO)n(C)n3)=O)CC2C)CC1=O 31579,C1(C(=O)NCC)Cc2nccnc2CN1C(c1ccc(F)cc1SC)=O 31580,CCC(C)C(O)C(C)C(=O)N1CCC(CCC(=O)NCCSCCOC)C1 31581,c1(C(=O)NC2CCN(C(CN(CCOC)C)=O)C2C)ccnc2[nH]c(C)nc12 31582,C12(C(=O)Nc3nccs3)CCC(CC1)NC2 31583,C(=O)(CC(F)(F)C(F)F)NC1C(NC(CC(n2c(C)cc(C)n2)C)=O)COC1 31584,C(=O)(C(C(C)(C)C)OC)N1CC(CNC(c2cc(CCC)[nH]n2)=O)(OC)C1 31585,C(=O)(C(C)(F)C(=O)NCCCOCCNC(C1(C)CCC1)=O)OC 31586,C1(OCC(=O)NCCC)CCN(C(=O)Cn2c(N)cnc2C)CC1 31587,c1(CC)noc(C)c1C(=O)NC1CC(n2cc(-c3ccc(CO)nc3)nn2)C1 31588,C(=O)(CCCCSC)NCC(CC)NC(=O)CSCC1CCCO1 31589,C=CC1CN(C(=O)C(CC(C)C)OC)CC1NC(=O)CCN1CCC(O)CC1 31590,Cc1cccc(C(C)C)c1C(=O)NCC1COCCN1C(C1CCNC(=O)C1)=O 31591,N1(C(c2c(CC=C)cccc2)=O)CC(C)CCC1CNC(=O)CN(C)C(N)=O 31592,c1(C(=O)NCC(CCOC)NC(c2cnc(CC(C)C)s2)=O)ccn(C)c(=O)c1 31593,c1(C(=O)NCCC(C)NC(C2(C(=O)OCC)CC2C)=O)noc2ncccc12 31594,c1(C(C(=O)NCCOC)N(C(C)COC)CC=C)ncn(C)n1 31595,c1(C(C(=O)NC2CC2)N(CCN=[N+]=[N-])CC)ccc(C2CC2C)o1 31596,C1(NC(CCN(S(C)(=O)=O)C)=O)C=CCN(C(c2n[nH]c(C)c2C(F)(F)F)=O)C1 31597,c1(OC)cc(C(=O)NC2CCCN(C(=O)CC(C)F)C2)c2ccccc2n1 31598,c1(C(C)C)cc(C(=O)NCC2(F)CC(NC(=O)CC(C)c3ccco3)C2)n(C)n1 31599,c1(NC(=O)CSCCC(O)c2cccs2)ccccc1COCC(F)(F)F 31600,C1(NC(c2nn(C)c3c2CCC3)=O)COC2(CCN(C(c3ncnn3C)=O)C2)C1 31601,C(=O)(CC1=NN(C)C(=O)C1)NC12CC(C(=O)NC3(C)C(C)C3)(C1)C2 31602,C1(C(=O)NC2C(NC(=O)COC3CC(F)(F)C3)CCCC2)CCC(F)(F)CC1 31603,CCCCC(C(=O)NC1(CO)CC(OC)C1)NC(=O)C(O)CC(C)C 31604,N1(C(c2c(C)cns2)=O)CC=CC(C(=O)NOCCOC(C)C)C1 31605,C1(CC=C)(NC(C2CC=CCC2)=O)CC2CCC(C1)N2C(C1CCCN1CC)=O 31606,C1(C(N(CCC#C)CCO)=O)CCN(C(c2occc2CC)=O)C(CC)C1 31607,c1(CN=C(NCC(O)CF)NC2CCC2)ccc2c(c1)CCO2 31608,c1(COC)cccc(C(=O)NCC2CCC(F)(CNC(=O)CC3CCCO3)C2)c1 31609,N1(C(CC2CC(=O)NC(=O)C2)=O)CCOC2(CCC(NC(C3CCSC3)=O)CC2)C1 31610,c1(C(N(CCNC(=O)C(F)=C2CCC2)C2CC2)=O)cc2ccc(Br)cn2n1 31611,c1(SCC(N2CC(OCCNC(C3(c4cccs4)CC3)=O)C2)=O)ccccn1 31612,c1(C(N2C(CN(C)C(C3CCCCC3)=O)COCC2)=O)cnc(S(C)(=O)=O)s1 31613,N1(C(CCSCC(C)C)=O)CCCC(C)(NC(=O)Cc2ccc(Cl)cc2)C1 31614,Cc1cc(CC(=O)NC(C)CNC(C2(c3cccc(Cl)c3F)CC2)=O)ccc1O 31615,C1(C(N(CC#C)CCF)=O)C(NC(=O)CCC2CC(OC)C2)C1(C)C 31616,C=CCCN=C(NCC1(OC)CCSC1)NC1CCCC(OC)C1 31617,N1(C(C(c2cnccn2)C)=O)CCc2[nH]nc(CNC(=O)C=CBr)c2C1 31618,c1(C(C)(C)C)ccc(C(=O)NC2(CNC(C3CCCOC3)=O)CCC2)[nH]1 31619,N12Cc3ccccc3CC1C2=O.c1(NC(C2C(N)C2)=O)cccc(C(=O)NC)c1 31620,c1(C(=O)NC2C(NC(c3cscc3F)=O)C2)ccc(-c2ccco2)[nH]1 31621,c1(CSCCN2CC(CNC(CC(C)C(F)F)=O)C2)cc(N)cc2ccccc12 31622,N1(C(C(=O)Nc2ccc(C)cc2)=O)CC2CCN(C(=O)Cc3cnc[nH]3)C(C2)C1 31623,c1(C(N(C)CC2CCCN2C(C2OCC2(C)C)=O)=O)c(C(F)(F)F)cnn1C 31624,CC(CC(=O)N1CCCOC(CNC(C2CC(F)(F)C2)=O)C1)C(F)F 31625,CC1(C)CC(CNC(c2ccco2)=O)CN1C(c1ccccc1C1CCCC1)=O 31626,C1(NC(C2CC(NC(COCC(C)C)=O)C2(C)C)=O)CCN(C)C1(C)C 31627,c1(OCCC)ccccc1C=CC(=O)NC(C)CC(C)NC(=O)CCSCC 31628,C(=O)(C(CNC(=O)CC1CCC(=O)NC1)C(C)(C)C)N1CC(CN(C)C)C1 31629,N1(C(CC2CCCN(C)C2)=O)CCN(C(=O)C(F)=CC2CC2)C(CC(F)(F)F)C1 31630,C1(OCC(=O)NC23C(CN(C(C4C(OC)CC4)=O)C2)C3)CCC(F)(F)CC1 31631,c1(C(C)(C)NC(=O)COC(F)(F)F)ccc(C2CC2)o1 31632,N1(C(c2cnccn2)C(=O)NCCSC)Cc2cc(Cl)c(Cl)cc2C1 31633,c1(C(=O)Nc2scc(CC(N3CCC(C(F)(F)F)C3)=O)n2)nc2ccccn2n1 31634,CC(C)CC(C(=O)NCC1(O)CC(O)C1)N(C)C(C1CCC1C#N)=O 31635,N1(C(CN(C)S(N)(=O)=O)=O)CCn2nc(CNC(C3(F)CCC3)=O)cc2C1 31636,C1(O)(CNC(c2cccn2C(F)F)=O)CCCN(C(=O)C=CCN2CCCC2)C1 31637,N1(C(N)=O)CCCCC1C(=O)NC1C=CCN(C(C2CCC2)=O)C1 31638,c1(CN)cccnc1.Cc1occc1COC(F)F 31639,C(CCC(O)C(=O)NCC(C)(C)C)NC(c1n(C)cc(Cl)c1)=O 31640,C1(C(=O)OC)(Cc2ncc(C(=O)NCCN3CCCC3)s2)CC=CCC1 31641,C1(C(C)C)C2CCC(C2)C1CN(CCCN(C)C)S(C)(=O)=O 31642,Cc1c(C(=O)N(C(C)CNC(=O)Cc2cnco2)C)cc(O)cc1N 31643,CC(C)CC(C(=O)NCCCNC(=O)C(C)(C)C1CCCO1)NC(=O)NC1CC1 31644,N1(C(CSCC=C)=O)CCC2(CC1)CN(C(C1C3CCC(C3)S1(=O)=O)=O)C2 31645,c1(COC(Cc2c(C)cc(O)cc2)=O)cc(=O)oc2cc(O)c(Cl)cc12 31646,c1(C(N2CCCC2CCCO)=O)ccc(-c2cccc(CNS(C)(=O)=O)c2)cc1 31647,c1(C(=O)NCC(CC=C)NC(c2cnn3cnnc3c2)=O)ncc2[nH]ncc2n1 31648,C1(NC(Cc2ccc(C)o2)=O)CC12CC(NC(C1(CF)CC(F)(F)C1)=O)C2 31649,CC1(F)CCCN(C(CC2CCCCCC2)C(=O)NC2CCOC2)C1 31650,C(=O)(C(C#N)C(C)(C)C)NCCc1c(C(N2CCC(CC#C)C2)=O)c[nH]n1 31651,C1(C(=O)NC2C(C)(C)C2)CCOCC1NC(=O)C(C)(F)c1ccon1 31652,Cn1cnc2cc(C(=O)NCC3(CO)CC3c3ccccc3)ccc2c1=O 31653,Cc1[nH]nc(C(N2CC3CCC3(NC(=O)C(F)=CC3CC3)C2)=O)c1[N+](=O)[O-] 31654,Cc1nc(N(CCCNC(c2cc(C3CC3)nn2C)=O)C)c(C)c(C)n1 31655,N1(C(C(C(=O)OC)C)=O)CCC(CNC(=O)C(=Cc2ccccc2Cl)C)CC1C 31656,c1(CNC(=O)Cc2cnco2)cccc(NC(=O)CC2CCSC2)c1 31657,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC(CC)CNC(=O)CNC(=O)CC(C)C 31658,c1(CC)[nH]c(C(=O)NC2CC(NC(=O)C#CC(C)C)C2)c(C)c1C(=O)OC 31659,N1(C(CCCc2cc(C)no2)=O)CCC2(CCCN(C(C3CCC(O)C3)=O)C2)C1 31660,c1(C(N(CCN(C(c2cc3sccc3[nH]2)=O)CC)CC)=O)c2ccccc2nn1C 31661,C=C(CNC(=O)C(F)C(C)CNC(=O)C=Cc1ccco1)C1CCOCC1 31662,c1(C(N2CC(NC(CC3N(C)CCC3)=O)C2)=O)ccc2c(O)nc(S)nc2c1 31663,C1(NC(C(C)OCC(C)C)=O)CCCCCN(C(=O)CCCC2CCCCC2)C1 31664,c1(-c2cn(C(C(N3CC(COC)OCC3)=O)C)nn2)ccnc(F)c1OC 31665,N1(C(C2C(C)=C2)=O)CCC(NC(=O)CN2CCCS2(=O)=O)CC1C 31666,c1(OC)cc(C(N2CCN(Cc3ccc(C)s3)CC2)C(=O)NC(C)C)ccn1 31667,N1(c2cc(NC(=O)OC)ncn2)CCC2C(CCN2CC2(c3cccs3)CC2)C1 31668,CN1CC2CC1CN2C(=O)CCC(=O)Nc1ccc(C(=O)NC(C)(C)C)cc1 31669,C(=O)(C1OCCn2ccnc21)NC1C(NC(c2cc(CO)on2)=O)C1 31670,N1(C(COCCC=C)=O)CCC(NC(c2nn(CC)cc2Cl)=O)C(F)C1 31671,C1(CNC(C2CC(=C)C2)=O)CCC2CN(C(c3ncoc3C3CC3)=O)CCC2C1 31672,c1(C(N2CCS(=O)CC(C)C2)=O)cccc2nc[nH]c12.Cc1cc2sc1c(=O)o2 31673,Cc1cnc(F)cc1C(N1CCN(C(=O)CCC[N+](=O)[O-])C(C)C1)=O 31674,C1(C(=O)NCCCOCCCC)CCC2(CC2)N1C(C1(SC)CC1)=O 31675,c1(C(N2C(C(C)(C)NC(c3cnn(C)n3)=O)CCC2)=O)ccccc1O 31676,C(=O)(C(C(C)C)NC(=O)CC1CCCCO1)N(CCC#C)CCOC 31677,C(CN(C)C)(C(=O)NC(c1ccccc1)C1C=CCC1)NC(C)=O 31678,C1(C(N(CC(CN(C(C(CC)C)=O)C)O)C)=O)CCC2CCCCC2C1 31679,Cc1ccc(F)c(C(=O)NCCCCN(C)C(C2(C)C=CCCC2)=O)c1Cl 31680,N1(C(c2cc(OCC)n[nH]2)=O)CC(C(=O)NCC(C)(C)COC)C(F)(F)C1 31681,c1(C(=O)NC(C2(O)CN(C(CC(C)OC)=O)C2)C)ccnc(C2CC2)n1 31682,C(=O)(C1CCCc2cc(O)ccc21)N(C1CCN(C(C2(C)CCCC2)=O)C1)CC 31683,c1(C2(C(N3CC(Cn4cc(CN5CCCCC5)nn4)C3)=O)CC2)ccc(Br)cc1 31684,C12CCCCCN1C2=O.N1(CC)CCN(C(C2CCCN2C(N)=O)=O)CC1 31685,C(=O)(CC1=CCCCC1)NC1COCCN(c2ccc(C(C)C)nc2Cl)C1 31686,O=C(C1CCCc2nn[nH]c21)N1CCC(OC2CN(CC(Cl)(Cl)Cl)C2)CC1 31687,C=CC1(C(=O)NCCC2CCOC2)CCN(C(=O)Cc2ccc(C)s2)C1 31688,C12(CC(=O)N(C3CN(C(=O)CN4C(=O)CCC4=O)C3)C)CCC(C)(C1)OC2 31689,C1(O)(C(=O)NCC(C)(C2CC2)NC(=O)CCN2CCC(O)CC2)CCCCCC1 31690,C1(NC(C2NC(=O)OCC2)=O)CCCN(C(c2cnc(S)n2C2CC2)=O)CC1 31691,O=C(CC(O)COC1CC1)NCC1(O)CN(C(=O)C(c2ccccc2F)O)C1 31692,C(=O)(C(C)(O)C(F)(F)F)NCC1(C)CCN(C(=O)Cn2ccnn2)CC1 31693,C(CC(=O)Nc1cc(C)cnc1C)(CC(C)C)NC(CC(COC)(C)C)=O 31694,N1(C(Cc2cc(C)sc2C)=O)CCCC(CO)(CNC(C2OCCC2(C)C)=O)C1 31695,Cc1ccc(F)c(CC(=O)NC2CC2NC(=O)CCCC2CC2)c1 31696,N1(C(C2C(=O)NCC2)=O)CCCC2(CCN(C(=O)CN3CCn4nccc43)C2)C1 31697,C(=O)(CC1C(=O)Nc2ccccc21)N1CCC(OCCCNC(COC)=O)CC1 31698,C1(NC(C(CCOCC)NC(=O)CS(=O)CC)=O)CCCC2(CC1)CC2 31699,c1(C(N2C3CC(N(C(C(CC)O)=O)C)CC2CC3)=O)c2ccccc2nn1C 31700,N1(C(CCC#C)=O)CC(C(=O)N(c2ncccc2C)CC)CC(F)C1 31701,c1(C(N2CCN(C(COCCC)=O)CC2)=O)cnc([N+](=O)[O-])cc1C 31702,N1(C(CC(C=C)(C)O)=O)CC(C2CN(C(C3CCC(C)(C)OC3)=O)C2)C1 31703,Cc1nc2c(s1)CN(C(c1ccc(N(C)C)cn1)C(=O)Nc1ccccc1C)C2 31704,C1(CC(=O)OCC)CN(Cc2nn(C)nc2Br)CC1(C)C 31705,C1(N(C(=O)Cc2csc(C(C)OC)n2)CC#C)CCN(C(C23CC(C2)C3)=O)CC1 31706,N(C(=NCC(C)C#N)NC(C)Cc1cccc(F)c1)C(C=C)C 31707,c1(CC(=O)NC2(CO)CN(C(CC(CC)C3CCC3)=O)C2)cnc2ncccn12 31708,C1(C(=O)NC2CCN(C(c3cc(=O)cc[nH]3)=O)C23CC3)CCc2nnc(O)n2C1 31709,c1(-n2cc(C3N(C(C(COC)NC(C)=O)=O)CCC3C)nn2)cccc(O)c1Cl 31710,C1(C(N2CC3C(NC(C4C=CCC4)=O)C(C3)C2)=O)COc2ccccc2O1 31711,N1(C(C(CC)NC(N)=O)=O)CCN(C(=O)CCc2ccc(Cl)nc2)CC1CC 31712,N1(CC(=O)N(CC(C)O)CC)CCN(C(c2cnncc2C)=O)CC1 31713,CCC(CN(C)C)CC(=O)NCCN(C(C1COCC2(CC2)O1)=O)C1CC1 31714,C1(C(=O)NC2CCC(CNC(C3(C)CC3C)=O)CC2)(NC(C)=O)CCCCC1 31715,N1(C(C(CC)C#N)=O)CC(C(=O)NCC2(O)CCN(C)C2)CC(C)C1 31716,c1(C(N2CC(C)N(C(c3cccnc3)=O)CC2)=O)cc2c(F)c(Cl)ccc2[nH]1 31717,C1(C(=O)NC(CC)C(C)O)CC(F)CN(C(c2ccc(C(F)(F)F)cc2)=O)C1 31718,C1(CNC(CSSC)=O)CCN(C(=O)C(C)Sc2ccc(N)cc2)C1(C)C 31719,c1(C(=O)Nc2nc(C3CCC(F)(F)CC3)cs2)ccc2c(c1)NS(=O)(=O)C2 31720,c1(C(=O)NC2CCCC(N(C(CCC(=C)C)=O)C)C2)cnc(O)c(OC)c1 31721,c1(CNC(c2n(C=C)ccn2)c2nnnn2CC2CC2)ccc2c(c1)OCCO2 31722,N1(Cc2cc(C(=O)OCC)on2)CC(NC(C2(CC)CC2)=O)CCC1C 31723,CCC(O)C(C)C(=O)NC1CCCCC1CNC(=O)CCCCc1ccccc1 31724,c1(C(=O)OC(c2ncc(Br)cn2)C)cc(Cl)c(N)c([N+](=O)[O-])c1 31725,c1(C(=O)NCC2N(C(C(C)n3ccnn3)=O)CC=C2)nn(C)c(Cl)c1Cl 31726,N1(C(C2(C)CCCCO2)=O)CCOC2(C1)CN(C(=O)Cn1ccnn1)C2 31727,C1(CCC(=O)N(CC(C)NC(C2CSC2)=O)C)CC(C)(C)CO1 31728,C(C)(C(=O)N1CC2(C)CC1(C(=O)NC1CC1C1CCCC1)C2)(C(C)C)OC 31729,C1(C(N2CC(CCNC(c3cc(C)oc3)=O)OC(C)C2)=O)CC1C1CCCCC1 31730,Cc1onc(C(F)(F)F)c1C(=O)NC1CCC(NC(=O)CC2CC(C)OC2C)C1 31731,Cn1nc(CNC(=O)C(C)(C)NC(C2CCCCN2C)=O)n(C)c1=O 31732,N1(C(C(C)C)=O)CC=CC1CNC(=O)CCC1(OCc2ccccc2)CCC1 31733,Cn1cc(CC(=O)NC2COCC2NC(c2cnns2)=O)cn1 31734,CC1CN(C(=O)Cc2cc[nH]n2)CC2(CCN(C(C3(O)CCCCC3)=O)C2)O1 31735,C(=O)(C(F)C(F)(F)F)N1CCC(N(CCC)C(c2nnc(S)n2C)=O)C1 31736,C12(NC(=O)CSCc3ccccc3)CCCC1N(C(=O)COc1cn[nH]c1)CC2 31737,C(CC1=CCCCCC1)NC(C(C)NC(C(C)NC(=O)C1CC1)=O)=O 31738,C(CCCC(=O)N(C(C)CCC(C)C)C)NC(C(COCC)C)=O 31739,c1(OC)c(C(=O)NC2CCN(C(c3cc(C(C)(C)C)[nH]c3C)=O)C2)ncnc1C 31740,c1(C(=O)NCC2CCC(NC(C3(CCCC)CC3)=O)C2)[nH]nc2ncnc(O)c12 31741,C12(Nc3c(C(=O)OCC)cccn3)CCCC1N(C(C1CCCSC1)=O)CC2 31742,N1(C(Cc2n(C)ccn2)=O)CCCC(C2CN(C(c3cc(Cl)ncc3F)=O)C2)C1 31743,Cc1ccc(C(=O)C(=O)NC2CC(NC(=O)C(C(C)C)N3CCN(C)CC3)C2)cc1 31744,C=C(C)C1CC(=O)N(C2CC2)C(C)C(=O)NO1.c1(C(N)=O)c[nH]ccc1=O 31745,c1(C(=O)NCC2N(C(c3cc(C)on3)=O)CC2)c(C)c(Cl)cc(C)c1N 31746,C1(N(C(COCC(=C)C)=O)C)CCCN(C(c2cscc2CC)=O)CC1 31747,C(C(=O)OCC)(C(C)C)NC(C(CC)C)=O.C1CC(=O)N1 31748,c1(C(=O)NC(CC=C)CNC(c2c(C)ncn2O)=O)cc(Cl)ccc1OC 31749,C(=O)(CC(C(F)F)NC(c1ccnc(C)n1)=O)NCCOCCC=C 31750,C1(C(=O)NCCN(CCCCCC)C(C23CC(C)C2C3)=O)CC=CCC1C 31751,N1(C(Cc2cnc(C)o2)=O)CC2CC(NC(c3ccc(C(C)(C)C)o3)=O)CC1C2 31752,CC1CCCn2ncc(C(N3CCC(NC(c4cc5ncccn5n4)=O)C3)=O)c21 31753,Cc1cccn2c(CC(=O)NCC3CC3NC(c3ccc(N)c(Cl)n3)=O)cnc12 31754,C12(C(N(CC(C)(C)NC(c3ccc(C)cc3F)=O)C)=O)CCOC1CCOC2 31755,C1(CNC(c2cc(OC)n(C)n2)=O)CC2(CC2)CN1C(=O)CCCc1cncs1 31756,Cc1oc2ccccc2c1C(N1CCCOC(CCNC(=O)C2=CCOC2)C1)=O 31757,N1(C(C(C=CC)O)=O)CCN(CC(=O)NCCC2(C)N=N2)CC1 31758,C(CN=C(NC(C)C1CC1)NC1CC=CCC1)n1ncc(C)c1 31759,N1(C(c2csc(C)n2)C(=O)NC(C(=O)OC)C)CCN(c2ccccc2O)CC1 31760,c1(C(=O)NCC=CCNC(c2c(Cl)cc(C)nc2)=O)c(C)nc(C2CC2)nc1O 31761,c1(CC)[nH]c(=N)sc1C(=O)N(C1CCCN(C(=O)CC2CCC23CCC3)C1)C 31762,CC1CN(C(C2CC23CC3)=O)CC(C)N(C(=O)C(C)Cc2ccccc2)C1 31763,C1(C(=O)NCC(CC(C)C)C)CN(C(C2CN(C)CC(C)O2)=O)CC12CCC2 31764,C1(CC=C)(C(N2CCSCC2)=O)CCCN1C(c1coc(SC)c1)=O 31765,c1(CC)cc(Br)cc(C(=O)NC2CCN(C(=O)Cc3nc[nH]n3)CC2F)c1N 31766,Cc1c(C(N2CCC(C)(NC(C34COCC(C3)C4)=O)C2)=O)cccc1Cl 31767,CC12CCOC(C(=O)NCC3CC(C(=O)NCCCN4CCC4)CO3)(C1)C2 31768,C1(CC)CN(C(=O)CCN(C(c2ccnn2C(F)F)=O)C(C)C)CC1O 31769,c1(SC)cn(C)nc1C(=O)NCC1CC(NC(C2CCC2C#N)=O)C1 31770,c1(N(C(C(N)=O)C2CCCO2)C)ccc2nc(O)[nH]c2c1 31771,c1(OC)ccc(NC(C2CC(NC(=O)COC(C)(C)C)C2(C)C)=O)c(O)c1 31772,c1(C(C)=O)cccc(OCC(N2CC(N(C(=O)Cc3ncc(C)s3)CCO)C2)=O)c1 31773,C(=O)(CC(O)CC(C)(C)C)NCC(CNC(CCCc1ccc(C)c(C)c1)=O)O 31774,c1(C(N(C)Cc2c(CNC(C3C(C)CCO3)=O)cccc2)=O)c(Cl)cncc1Cl 31775,c1(C(=O)NCCOCCCNC(CCCC(CC)C)=O)c(F)ccc2n[nH]cc12 31776,C1(C(=O)NCCC2(O)CN(C(C3COC4(CCC4)C3)=O)C2)CCCCC(F)(F)C1 31777,Cc1cc([N+](=O)[O-])cnc1N1CC2CCN(C(=O)Oc3ccccc3)CC2C1 31778,C1(N(C(C(C2CCCC2)NC(C)=O)=O)C)CCN(C(c2ccc(CO)s2)=O)C1 31779,c1(CC(N2CC(CC=C)(NC(=O)CC3CCC(O)C3)C2)=O)sc(C)cc1C 31780,Cc1cc(C#N)cnc1C(=O)NC1(C)CCCN(C(=O)Cc2cccnc2Br)C1 31781,C12(C(=O)NC(CNC(c3ccnc(C)c3C)=O)(C)C)CCOC1CCOC2 31782,N1(C(COC2CCN(C(CC3CCCN(C)C3)=O)C2)=O)CC2CC2C2CC12 31783,C1(C(=O)NCC2(NC(Cn3c(N)cc(C)n3)=O)CC2)CN(C)CCN(C)C1 31784,C1(NC(C2CC(C)NC(=O)C2)=O)CN(C(=O)CC2CC(F)(F)C2)CC12CCCC2 31785,C(=O)(C1(C)c2ccccc2-c2ccccc21)N1CCC(CC(=O)NCCCOC)C1 31786,C#CCCCC(=O)NCC1CC(NC(=O)CC2(OC3CCCCC3)CC2)C1 31787,c1(C(N(C2CN(C(C(C)OC)=O)C2)C)=O)c(NC(C)=O)c[nH]c1C 31788,c1(C(=O)NC(CN(C(=O)CC2CCC(=O)NC2=O)CC)C)cc(O)cc(C#N)c1 31789,CC1CN(N(Cc2ccc(F)cc2Cl)Cc2ccncc2)CC1F 31790,N1(C(C(C(C)OC)N(C)C)=O)CCC(C)C(CC(N2CC(F)(F)CC2CO)=O)C1 31791,CCC(C)C(CC(=O)N1CCC(F)(F)CC1C)NC(c1n[nH]c(=N)[nH]1)=O 31792,CCCC(CC)CC(=O)N1CC(CNC(c2cc(Cl)ccc2C)=O)C2(CC2)C1 31793,C1(CN(C(C(C)n2cccn2)=O)C)CN(C(c2cc(O)n(C)n2)=O)CC12CC2 31794,C(CCCC(C)(F)F)(C(=O)NCC1CCCO1)N(C)CCN1CCCC1=O 31795,CCC(CC)C(C)C(=O)N1CCC2(CC2C(=O)N(C(C)CO)CC)C1 31796,C1(NC(C(C(=O)OC)OC)=O)CCN(C(C2CCOC2)=O)CC1F 31797,C(COC(C)=O)(C(=O)N(C)CCN(C(=O)CCCOC(C)(C)C)C)NC(=O)OC 31798,C#Cc1ccc(C(=O)NCC(O)CCNC(=O)C(C)(CC)C(=O)OCC)c(C)c1 31799,CCC(CN(C)C(c1cscn1)=O)NC(=O)C(C)C1CCCC1 31800,Cc1ccc(C(=O)NC2C(Cl)(Cl)C23CC3)cc1Br 31801,N1(C(C(C)CC2CCCCC2)=O)CCC(O)C(NC(=O)C=CC2CC2)C1 31802,C(C(C)(F)C(F)(F)F)NCc1c(CNC(=O)OC(C)(C)C)cccc1 31803,C12(NC(COCCCCOCC#C)=O)CCC(CN(C(c3cc(C)cs3)=O)C1)C2 31804,C1(C(=O)NCCOCCC=C)(CNC(C2CC2=C)=O)CC(=C)C1 31805,Cc1cnc(F)cc1NC(=O)NC1(CN(C)C)CCN(C)CC1 31806,c1(C(=O)NC(C2CCOC2)CNC(c2ccc(C)nc2)=O)c[nH]cc(F)c1=O 31807,C(=O)(CC1=NNC(=O)C1)N1C2CN(C(C(c3cccc(C)c3)O)=O)C(C2)C1 31808,c1(C(N2CC(CC(N3CC(C#N)C3)=O)C3(C2)CC3)=O)c[nH]c2ncccc12 31809,c1(C(N(C(CNC(Cc2c(C)ccc(F)c2)=O)C)C)=O)cccc(S(C)=O)c1 31810,CCC(C(=O)NCc1cnn(C)c1C(=O)NCCN(C)C(=O)C1CC1)C(F)(F)F 31811,Cc1ncc(N)cc1C(N1CC(C2(NC(=O)Cn3cc(Cl)cn3)CC2)C1)=O 31812,C1(C(N2CCC(CC=C)C2)=O)N(C(C2COCCO2)=O)CCC1(C)C 31813,CCC(CC)CC(=O)NC1CC(C(F)C(=O)Nc2c[nH]ccc2=O)C1 31814,Cc1cc(C(=O)NC2CCC(CC(=O)NC3(C4CC4)CCCC3)CC2)ccc1O 31815,C1(NS(CC)(=O)=O)CCCN(c2nnc(-c3nn(C)cc3Br)n2C2CC2C)C1 31816,c1(OC)cccc(NC(C2(O)CCN(C(c3ccc(O)c(F)c3)=O)C2)=O)c1C 31817,N1(C(C23CC(NC(c4c(CCC)nco4)=O)(C2)C3)=O)CCC(O)CC12CC2 31818,CCC(O)CC(=O)N1CCCCC1Cn1cc(C2C3CCCCC23)nn1 31819,N1(C(C(C)NC(=O)OC)=O)CCN(C(=O)Cc2cccnc2C)CC(C)(C)C1 31820,c1(CC(=O)NC23CCC(C2)N(C(=O)C(F)n2ccnc2)C3)cc(F)cc(F)c1 31821,N1(C(CC2CC(SC)C2)=O)CC(F)(F)CC1CCNC(=O)CSc1nncn1C 31822,C1(CCN(C(=O)COC(c2ccccn2)=O)C)CCCCN1C(=O)C(C)(C)C 31823,CCC(CC)C(=O)N1CC(C(=O)NCCNC(C2CCNC(=O)C2)=O)C1 31824,N1(C(c2n(C)ccc2)=O)CCC(OC2CN(C(C3(C)CC=CC3)=O)C2)CC1 31825,c1(CCC)nc(C)c(CN2CCC(N(C)C(C3CCOC(C)C3)=O)C2)o1 31826,c1(CC)ccc(C(=O)Cc2ccccc2)cc1C.C12CN(CC(OC)C1)C(=O)N2 31827,N1(C(C(c2nccn2C)OC)=O)CCC(O)(CNC(c2scnc2CO)=O)CC1 31828,C(=O)(C(F)C(C)(F)F)NCCCN(C(CCC(=O)NCCCN(C)C)=O)C 31829,N1(C(c2nc(C)oc2)=O)CC(CCNC(C2CC3C=CC2C3)=O)C(C)C1 31830,C1(NC(C(CC)OCC)=O)CC2(C1)CC(CNC(c1cn(CC)nn1)=O)C2 31831,C1(C(N(CCCC(=O)NCCOC(C)C)C)=O)CCCC(C)C1 31832,C1(NC(C(CCO)N(C)C)=O)CN(C(C2CCC=CCCC2)=O)C2(CCC2)C1 31833,c1(OCC)cc(C(=O)N(CC(O)CNC(=O)CCc2cc[nH]n2)C)on1 31834,N1(C(C)C)CC(C)C(c2nnnn2C2CCCC2)(NC2CC2)C1 31835,C1(NC(C(C)OCC#C)=O)CCN(C(c2cnc(C(C)(C)C)nc2)=O)C1C(C)C 31836,c1(C(=O)NCC2CCN(C(C3CCC(CC)O3)=O)CC2C)csc(=NC2CC2)[nH]1 31837,C1(SCc2cc(CC)n[nH]2)CCN(C(=O)CN(C)CCc2noc(C)n2)CC1 31838,N1(C(C=CCC)=O)CCC(C2CC2)(CNC(c2ccc(Cl)s2)=O)C1 31839,Cc1ccn(C)c1C(=O)NC1CC1NC(C1(C2CCCCC2)CCOCC1)=O 31840,Cc1cccnc1CNC(C1COCCC1NC(=O)COC(C)C)=O 31841,N1(C(c2cc(C3(C)CC3)n[nH]2)=O)CCC2(CCC(NC(C3(CO)COC3)=O)C2)C1 31842,C(=O)(C1CCc2c(Cl)cccc21)NC(C)CNC(c1ccc([N+](=O)[O-])cc1F)=O 31843,c1(C(C)(C)C)ccoc1NC(C1(NC(=O)CSC2CCCCO2)CCCC1)=O 31844,C1(NC(CC2CC(C)C(C)CC2)=O)CC2(C1)CC2N=c1cnc(F)c[nH]1 31845,C1(CC)CN(CC)CCN1C(C1C(CNC(=O)C#CC(C)C)C1(C)C)=O 31846,CCCCC(C(=O)NC1CC(CCF)C1)NC(=O)C=CCCC(C)C 31847,C1(NC(C2CC2CF)=O)CC2CC1N(C(=O)Cn1ccccc1=O)C2 31848,CC1N(C(c2cc(CNC(c3cc(CO)on3)=O)[nH]n2)=O)CCOC1(C)C 31849,c1(C(=O)NCC(CC)NC(=O)C(C(C)C)N(C)C)cc(Cl)ccc1[N+](=O)[O-] 31850,C1(C(=O)NCCCN(CCCNC(C2(C)COC2)=O)C)CCCC1S(C)(=O)=O 31851,C1(C(=O)NC(C(=O)OC)C(C)C)CC12CCN(C(=O)C(O)C(F)(F)F)C2 31852,N1(C(C(CSC(C)(C)C)NC(C)=O)=O)CC2CC(NC(=O)CSC(F)(F)F)C(C2)C1 31853,CCC(C#N)C(=O)N1CCCC1NC(=O)C(C)CN(C(=O)OC(C)(C)C)CC 31854,N1(C(CCC=C(C)C)=O)CC(F)(F)CC1C(=O)NC(c1ccc(C)s1)C 31855,c1(C(N2CC(NC(C3C(OC)CC3)=O)C(O)C2)=O)sc2sccc2c1Cl 31856,c1(NC(=O)NC2CC2C(=O)Nc2ccc(CO)cn2)ccc(Br)cn1 31857,C(C)(C(CC(=O)NCc1ccc(C#N)s1)NC(C1CCC(C)(C)C1)=O)OC 31858,C(=O)(C(C)(C)C(=O)N(C)C)NC(CNC(CSCC#C)=O)CCOC 31859,n1(CC)cc(C(N2CCN(CCO)C(C)C2)=O)c(=O)c2cc(Br)ccc12 31860,c1(C(=O)NCCCN(C(c2n[nH]cc2Br)=O)CC)nccc2ccn(C)c12 31861,c1(CC(=O)NCCC(=C)CNC(=O)Cc2ccc(C)c(C)c2)ccc(C)c(C)c1 31862,CC(C)CC(F)(F)C(=O)NC1CC2(C1)CC2NC(=O)CCN1C(=O)CN(C)C1=O 31863,C(CCCCC(=O)N1CCCC1C(=O)Nc1cncc(C(=O)OC)c1)NC 31864,C1(N(C(c2c(SC)cccc2)=O)C)CCN(C(c2c[nH]c(C#N)c2)=O)CC1C 31865,c1(C(=O)NCC(=O)NC2CC2)ccc(C(=O)NC2CC(C(F)(F)F)C2)cc1 31866,CC1CCN(C(c2ccnc(-n3cccc3)c2)=O)C1CNC(=O)C(C)CO 31867,C(CC(C(=O)NCc1ncc(C(N2CCC(C)(C(N)=O)C2)=O)cn1)OC)OC 31868,C(CC(=O)NCCCCCNC(C1CS(=O)(=O)C1)=O)(C1CC1)NC(=O)OC(C)(C)C 31869,Cc1ccncc1CC(=O)NCC1(C)CCC(NC(=O)CCc2cccs2)C1 31870,c1(C(N2CCC(C)(NC(C(C)NS(CC)(=O)=O)=O)C2)=O)ccc2c(c1O)CCC2 31871,C1(C(N2CCC(NC(=O)OC)CC2)=O)CN(C(=O)Cc2cn[nH]c2)CCC1(C)C 31872,N1(C(C(C)C2CCC2)=O)CC(CC(=O)NC2CCCCCC2F)CC1(C)C 31873,c1(C(=O)NC(C2(CNC(CCOCCOC)=O)CC2)C)cnc(C)s1 31874,c1(OC)ncc(-c2cncc(C(=O)NCC3CCC(CO)CC3)c2)c(SC)n1 31875,c1(CC(=O)NCC2CCCN(C(=O)C(c3ccc(F)cc3)O)C2)cccnc1Cl 31876,O=S(=O)(C1CCC(c2ccccc2)CC1)NCCNCc1cccnc1 31877,CC(C)CC(O)CC(=O)N1CCCCCC1C(N1CC(N(C)C)C1)=O 31878,c1(C(=O)NCC(C)CNC(c2c[nH]cc(Cl)c2=O)=O)cccc2c1oc(=O)n2C 31879,C1(NC(COCCC=C)=O)CCCCCC1C(=O)Nc1cc(C)ccc1OC 31880,C(=O)(C1OC(=O)c2ccccc21)N1CCC2(C(NC(c3c(C)occ3)=O)C2)CC1 31881,C1(CC(=O)NCC(C2CCN(C(C3CNC(=O)N3)=O)CC2)C)CCCCCC1 31882,CC(C)CC(C(=O)NOC1CCOCC1)ONC(=O)CNc1ncccn1 31883,CC(C)C(O)C(=O)NC1(c2ccccc2)CCN(C(=O)Cc2csc(Cl)c2)C1 31884,C1(CCCCCNC(c2cnccn2)=O)CCN(C(C2CCC(F)C2)=O)CC1 31885,CS(=O)(=O)c1ccc(C(=O)NC2CC23CCN(C(C2CCCSC2)=O)CC3)s1 31886,c1(C(=O)NCC2OCC(=O)NC2)n[nH]c2ccc(-c3c[nH]c4nccc-4c3)cc12 31887,c1(C(=O)NCC(CC)NC(=O)CSc2nnnn2C)cccc(N2CCCC2)n1 31888,CCC(CCCC(=O)NCCN(CCO)CC)NC(c1nc(C)c(C)s1)=O 31889,CC1CNC(=O)CN1C(C1CC12CCN(C(=O)CN1CC3CC3C1)C2)=O 31890,N1(C(C(CC)CCOC)=O)CC2CC(C1)C(CO)C2NC(c1csc(CO)n1)=O 31891,N1(C(C2CC(=C)C2)=O)CCC(C2(NC(=O)Cc3cnccn3)CC2)CC1 31892,Cc1nsc(N2CC(F)(F)CC2CNC(c2cn(C3CCC3)nc2C)=O)c1C#N 31893,c1(COC(N2CCN(C(CC(C)C)=O)CC2)=O)cccc2c1OCCC2CCO 31894,N1(C(Cc2ccc(C)s2)=O)CCC2C(C1)CN2C(=O)Cn1cc([N+](=O)[O-])nc1C 31895,C=C(Cl)C(C)(C)C(=O)N(CCCNC(C1(C(F)(F)F)CCCCCC1)=O)C1CC1 31896,CC(CC(F)(F)F)C(=O)N1CCC(C(=O)NCc2cc(O)ns2)C12CCC2 31897,C1(C(=O)NCC(C)CN(C(=O)CSCc2cccnc2)C)C2COCC12 31898,c1(CCC)cnnc(C(=O)NC2CCC2NC(=O)CCC(C)C)c1 31899,c1(C(=O)NC(CNC)C(C)(C)C)cc2cccnn2c1 31900,N1(C(C(CC)Cl)=O)CCCC12CCCN(C(=O)CC(C)C)CC2 31901,C1(CC(N)=O)(NC(=O)CCN2CCC(F)(F)C2)CCCN(C(=O)CC2CCC2)C1 31902,C12(CNC(c3ccsn3)=O)CCCC1CN(C(C13CCC(CF)(C1)OC3)=O)C2 31903,C1(CNC(=O)COCC2CC2)CC(NC(C2(C(F)F)CCC2)=O)C1 31904,CCC(C)(CC)CN=c1nc(N2CCC(n3cncn3)C2)c2[nH]ccc2[nH]1 31905,N1(C(CCNC(=O)OC)=O)CC(C)(NCC2=NOCC2)CC1(C)C 31906,C(C(F)(C(=O)NCCC(O)C(C)C)C(C)C)NC(C(=Cc1ccccc1)C)=O 31907,C(=O)(C(O)CCCNC(=O)CC=Cc1ccccc1)N(C1CCC(C)(CN)CC1)C 31908,C(=O)(C1COc2ccccc21)NC1CN(C(CC(CC)OC)=O)CC2(C1)CC2 31909,N1(C(CC2C(C)(C)C(NC(=O)CCCC3CCC3)C2)=O)CCC2(CC1)CC2C#N 31910,N1(C(C=CC)=O)CCC(C2CCC2)(CNC(=O)CC=C(Cl)Cl)CC1 31911,C1(C)(C(=O)NC2(CNC(C(COC)(C)C)=O)CCCCCC2)CC(C)OC(C)C1 31912,C1(NC(c2ccc(F)s2)=O)CC(O)CN(C(=O)C2=CCCS2)C1 31913,CCC(C)C(C)C(=O)NCCCN(C(c1ncc(C)cn1)=O)C1CC1 31914,c1(C(C)=O)cc(NC(C2(F)CCN(C(c3ccc[nH]3)=O)CC2)=O)ccc1F 31915,C(C1CN(C(=O)C(C)C2CCC2)CC1C(=O)NC(C)C(F)(F)F)=CC 31916,c1(N(CCCCC=C)C)nc(N2CCCC(C)C2)c2c(n1)CSC2 31917,C(=O)(C(CCC1CCC1)NC(c1cnc(C2CC2)o1)=O)Nc1c(C)csc1 31918,N1(c2nc(C)cc(OCC)n2)Cc2nccn2CC(NC(c2coc(C)c2)=O)C1 31919,Cc1ccc(O)c(C(=O)NC2CC(OCC(N3CCCC(F)(F)C3)=O)C2)c1 31920,c1(C(=O)NC(CNC(c2c(C)ccnc2)=O)(C)C(C)C)onc2c1CCCC2 31921,CC(C)(C)C(O)CNC(=O)NCC(COC(=O)Nc1ccccc1)(C)F 31922,S(=O)(=O)(c1ccc(Br)cc1N(CC(CC)OC)C)N(C(C=C)COC)C 31923,CC1CC(NC(c2coc(O)n2)=O)CN(C(=O)CSc2nncn2C(C)(C)C)C1 31924,C(=O)(C=C1SCC(=O)N1C)N1CCC(NC(c2c(C)c(Cl)sc2Cl)=O)CC1 31925,Cc1nc2cc(C(=O)NCC3CN(C(C4CCOC4)=O)CC3C)cc(Br)c2o1 31926,Cc1noc(C(=O)OCC(=O)NC2CCC(C)(C)C2)c1I 31927,Cc1cc(C(N2CCN(C3COCC3NC(=O)CC3(C)CC3)CC2)=O)oc1C 31928,N1(C(C2CC=CC(NC(CCCC)=O)C2)=O)CC2(CCNC(=O)O2)C1 31929,CCC(C)CC(=O)C(=O)N1CCCC(CN(C)C(c2cc(O)n(C)n2)=O)C1 31930,N1(C(C=C(CCC)C)=O)CC(NC(=O)CCCn2cccc2)CC12CCC2 31931,C(=O)(C(C(C)CC)c1ccco1)NC1(CCNC(CCC)=O)CCCC1 31932,Cc1cc(C(N2CCOC(CCNC(C3CC(C)(F)C3)=O)C2)=O)n2nccc2n1 31933,C1(C(C)NC(Cc2c(C)cco2)=O)CCCN(C(=O)CCc2c(C)noc2Cl)C1 31934,N1(C(Cc2cccc(C#C)c2)=O)CCN(C(=O)CC(C)(C)C=C)C(C)C1C 31935,CCC(CCCC(=O)NCCCc1nncs1)NC(C1CCC(O)C1)=O 31936,c1(C(=O)NCCCN(C(=O)CC2CCN(C)C2=O)CC)cc(OC)c(Cl)s1 31937,N1(C(C2Cc3ccncc3C2)=O)CC2CCN(C(c3ncccn3)=O)C2C1 31938,CC1(C)COCCC1C(N1CC2CC(NC(c3cnoc3C3CCC3)=O)C2C1)=O 31939,c1(C(N2C(CNC(CCOCC(C)C)=O)CC3(CC3)C2)=O)nsc2ccccc12 31940,c1(CCC)ccc(N)c(C(=O)NC(CNC(c2cc(O)n(CC)n2)=O)CCC)c1 31941,n1(CC)nncc1C(=O)NC12CC(CNC(=O)C(C3(O)CCCC3)F)(C1)C2 31942,C1(CCC)CCC(NC(=O)C(Cn2ccnn2)NC(=O)CC2CCOCC2)CC1 31943,c1(C(=O)NC(CNC(c2c(C)nn(C)c2C(F)(F)F)=O)C)ccc(C#N)nc1O 31944,c1(CN2CCC(N(C)C(c3c(I)ccnc3Cl)=O)C2)cc(F)ccc1[N+](=O)[O-] 31945,c1(NC(C2C(NC(C3C(C)(C)OC(=O)C3)=O)C3CCC2C3)=O)cc[nH]c2nccc1-2 31946,Cc1cccnc1C(=O)NCC1(C(=O)NCC(c2nccs2)C)CC2(CC2)C1 31947,n1(C(C)C)ncc(F)c1C(=O)NC1CCCC1CNC(=O)C(c1ccccc1)C 31948,C1(CNC(CCN(C(=O)C(C)NC(N)=O)CC#C)=O)CC2CC1CC2O 31949,N1(C(C2(SCC)CCC2)=O)CCC(N(C(=O)Cc2cccc(CO)c2)CC)CC1 31950,Cc1cnc2n1CCC(C(=O)NCCNC(=O)C1=CCCS1)C2 31951,N1(C(C23OCC(C)(C2)C3)=O)CC=C(CNC(=O)Cc2cccnc2)CC1 31952,N1(C(c2ccnc3c2CCC3)=O)CCN(C(C2CCC(O)C2)=O)C2(CCC2)C1 31953,C1(NC(COCCCC)=O)CC2CCC(C1C)N2C(C12CC(CO1)C2)=O 31954,c1(NCC2CN(C(C3CCc4nccn4C3)=O)C2)ncc([N+](=O)[O-])cc1F 31955,CC1CCN(C(=O)CN2CCCCCC2)CC1NC(=O)CC1CC=CCC1 31956,CC(CC(=O)N(C)CC1CCCN(C(C23CCC(C2)C3(C)C)=O)C1)CC(C)(C)C 31957,c1(CC(=O)N(C(CCNC(C(COC)COC)=O)C)C)cnn2ccccc12 31958,C1(OCCCNC(C(C)c2ccsn2)=O)CCN(C(c2c[nH]ccc2=O)=O)CC1 31959,CCCC(C)(O)C(=O)NCC(CO)NC(c1ccnc(Cn2cnnc2)c1)=O 31960,N1(C(C2CCC(=O)CC2)=O)CCC2CCCC12C(=O)NOCC1CCOC1 31961,C(=O)(C(C)(C)C(N)=O)N1CCC(CN(C(=O)CC2SC(=N)NC2=O)C)CC1 31962,C1(CC(N2CC(C)(NC(=O)CCCC3CCOCC3)C2)=O)CCCCC1O 31963,N1(C(c2cc(N)cc(F)c2)=O)CCC(C2CC2)(CNC(c2ccc(CO)o2)=O)C1 31964,CC(C)CCCC(C)C(=O)N(C1CCN(C(=O)C=CCO)CC1)CC1CCCO1 31965,c1(C(=O)NC23CC2CN(c2ncc4sccc4n2)C3)cc(Br)cc2[nH]ccc12 31966,Cc1ncccc1CC(=O)NC1CC(NC(=O)CC2COC(C)(C)C2)C1 31967,C1(OCC(N2CCN(C3CC(C)OC3=O)CC2)=O)CCC(F)(F)CC1 31968,C(CC(CC)C(=O)N1CCN(C(=O)Cc2ccc(CC)cc2)CC1)=CC 31969,C(CCS(=O)(=O)OC(C)(C)C)OC.c12ncn(n1)CNCCOCCN(C)C2=O 31970,c1(C(=O)NC2(C(F)F)CC(NC(c3ccc[n+]([O-])c3)=O)C2)cnc2n1CCCC2 31971,c1(C(N2CC3CN(C(c4scc(OC)c4)=O)C3CC2)=O)[nH]cc2c1CCS2(=O)=O 31972,CC(=O)C(C)CC(C)C(=O)N1CC=CC1(C)C(=O)N(C1CC(C)(C)C1)C 31973,N1(C(C2(SC)CC2)=O)CC2CC1CC2NC(=O)Cc1c[nH]nc1C 31974,c1(C(=O)NCCC2(C(NOCC=C)=O)CC2)ccc(C#N)c(C)n1 31975,c1(CCC(N2C(C)C(NC(C3(CO)CC3)=O)CCC2)=O)ccc2c(c1)OCCO2 31976,C1(NC(=O)C=CC2CC2)C2CCN(C(=O)C=CCOc3ccccc3)C12 31977,c1(CC(=O)NCC2N(C(C(CCOC)C)=O)CC=C2)cn2c(C)csc2n1 31978,N1(C(C(C)OCC#C)=O)CCCC1C(C)(C)C(=O)N(C)CCN(C)C(=O)C1CC1 31979,Cc1ccnc(C(=O)NCC(C)(C)CCNC(=O)CN2CCOCC2)c1 31980,N1(C(c2c(C(C)C)scn2)=O)CCC(C(C)(O)CNC(C2CCCO2)=O)CC1 31981,c1(C(N2C(CNC(Cc3ccc(C)cn3)=O)CC2)=O)cc(N)ccc1C 31982,c1(C(N)=O)ccc(NC(=O)CC2CN(C(c3ccc(Br)s3)=O)CCO2)cn1 31983,c1(NC(CC2N(C(C(CC)=O)=O)CCOC2)=O)nc(O)ccc1[N+](=O)[O-] 31984,C1(C(C(=O)N(CCC(=O)NC(c2ncc[nH]2)C)C2CC2)C)CCC(=O)N1 31985,C1(CC)(CNC(=O)C(Cc2ccoc2)NC(=O)CSCCC#N)CCCC1 31986,C(CC(C(=O)NC1(C)CC1)NC(=O)C=CC1CCCN1C)N(C)C 31987,c1(CC)ccc(C(=O)NC(C)CCN(C)C(C2CCOC2C(C)C)=O)o1 31988,N1(C(C(C)OCOC)=O)CC2CN(C(=O)C(C3CCCCC3)C)CC2(C)C1 31989,CC1CC(CNC(C2(C(F)F)CC2(F)F)=O)=NO1 31990,c1(N2C3(CNC(N4CCC5(CCOC5)C4)=O)CC3CC2)ncnn2ccc(Br)c12 31991,CC(CC1CCC1)N=c1[nH]c2c(c(=NCC3C4CCCC34)[nH]1)CSC2 31992,c1(C(=O)NCC(C)N(C(c2cc(C)n(C)n2)=O)C)ccc2ccccc2c1O 31993,Cc1nn2c(c1C(N1CCCC(NC(c3ccc(CO)s3)=O)C1)=O)CCCC2 31994,C(=O)(C(O)CC1CC1)NC(C1CCCC1)CNC(=O)Cn1cnnn1 31995,c1(C(C)C)ccc(C(CNC(C2CC(C)(C)C2)=O)NC(=O)Cn2ccnn2)cc1 31996,C1(NC(C(C)OCCN(C)C)=O)COCCC1NC(=O)Cn1cnnc1O 31997,C(=O)(C(C)S(=O)(=O)C(C)C)N1CCC(NC(c2cc(C)c(OC(F)F)cc2)=O)C1 31998,Cc1cc(C(=O)NCCOc2ccc(F)c(F)c2)c2ccc(Br)cc2n1 31999,C(=O)(CCCCSC)NC1(CNC(C(C=C)OC)=O)CCCC1 32000,c1(C(=O)NC2(CO)CN(C(C(C)SCC)=O)C2)cc(OC)cc2c1OCC2 32001,C(=O)(CC(F)(F)C(F)F)NCC(CC=C)C(=O)N1CC2CC2C1 32002,C1(CCNC(C2CC(C)(F)C2)=O)CCN(C(c2ncoc2-c2ccco2)=O)CC1 32003,C(=O)(C(C)CC(F)(F)F)NCCCC(C)NC(C1(N2CCOCC2)CCCC1)=O 32004,N1(C(c2ncc(Br)s2)C(=O)NC2CC(C(=O)OC)C2)C(C(N)=O)CC2CC12 32005,C#Cc1cncc(C(=O)NCC2(O)CC(CNC(c3ccc(C)c(C)n3)=O)C2)c1 32006,C1(C(=O)NCCCN(C(=O)C(O)c2cnc[nH]2)C(C)C)CCC(OC(F)F)CC1 32007,C1(NC(C(CC=CCC)C)=O)COCCN(C(=O)CCCCCOC)C1 32008,C1(C(N(CCCCCNC(=O)CCCn2ccnc2)C)=O)CC2CCC1C2 32009,C1(NC(C(CCOC)OC)=O)CCCCC12CCN(c1ncnc(C)c1F)CC2 32010,N1(C(C(CC)N(CC2(OC)CCCCC2)CC)=O)CCC=C(C(=O)NCCO)C1 32011,c1(C(=O)NC(C(C)NC(C(COC)C)=O)CO)c(C)ccc(Cl)c1N 32012,c1(C(C(=O)NCCCC2CC2)N(C(C)C2CC2)C)ccc(C(F)F)cc1F 32013,C1(C(=O)NC2(CNC(c3cc(Cl)c(Cl)[nH]3)=O)CCC2)CCCC(F)(F)C1 32014,CCC1=NOC(CC(=O)NC2CCCC2NC(c2cnc(CC(C)C)[nH]2)=O)C1 32015,c1(N(C)C)cccc(N2CCN(C(N3CC(SC(C)(C)C)OCC3)=O)CC2)c1 32016,N1(C(C(CC)C#N)=O)CC(C2CCCN(C(c3nc(OC)c(C)s3)=O)C2)C1 32017,CCC(CC(C)C)C(=O)N1CCC(C2CC2)C1CNC(=O)CC1CC1(Cl)Cl 32018,C1(C(N2CC(C(N3CCC(CCN(C)C)C3)=O)(CC)C2)=O)COCC(C)O1 32019,c1(C(=O)NC2C3CN(C(C4C(C)=NNC4=O)=O)CC2C3)cc2cccc(C)c2o1 32020,c1(NC(C2CCC(CNC(C3CC3(Cl)Cl)=O)O2)=O)cncc(F)c1 32021,C(CCCCNC(=O)CCC1(N(C)C)CCC1)N(C(=O)CC1CC1(C)C)C 32022,CC1(C)CCC(C(=O)NCc2ncoc2CNC(=O)CC2CC3CCC2C3)CC1 32023,C=CCN=C(NCc1nnc(C(C)C)s1)N1CCC(OCC(C)C)C1 32024,C(=O)(C(CCC(C)C)NC(=O)C(=C1CCCCC1)F)NC(C#C)C(C)C 32025,n1(C(=O)NCC23CC(CN2C(=O)COCC2CC2)C3)cc(Br)c(O)nc1=O 32026,n1(CC)nc(C(=O)N(C(C)CCNC(=O)C(C)CSC(F)(F)F)C)cc1O 32027,Cc1oc(C(C)C)nc1C(=O)N(CC(O)CN(C(=O)C=Cc1ccncn1)C)C 32028,c1(C(N2CCSCC2c2ccc(Cl)cc2)=O)cnc2c[nH]nc2c1 32029,C1(NC(c2ccon2)=O)CCC2CCN(C(=O)C#CC3CCCCO3)C1C2 32030,N1(C(C(CN(C)C)O)=O)CC(C)C(C)(C(=O)NC2CC(CC(C)(C)C)C2)C1 32031,C(=O)(C1CCCc2scnc21)NCC1CN(C(CCCCC(=O)NC)=O)CC1C 32032,CCCCCC(C)CC(=O)N1CC=CC(NC(C2(C)CC3(CCC3)C2)=O)C1 32033,C(=O)(CC1=CCCC1)NCc1c(CNC(C2C(=O)NCC2)=O)cccc1 32034,C(=O)(CC(C)C(=O)NC1C=CC(CC(=O)N(C2CC2C2CC2)C)C1)OCC 32035,C1(COC)CC2(CCN2C(=O)CC2CCN(C(=O)C(C)Cn3cccn3)C2)C1 32036,C1(CNC(C2(C=C)CC2)=O)CC(C(C)(C)C)CCN1C(=O)C(=CC1CCCC1)C 32037,N1(C(C(CC(C)C)F)=O)CC2CCN(C(c3cnn4ccsc34)=O)CC12 32038,c1(C(CNC(C2C(C)C2)=O)NC(c2cccc(C3CC3)c2)=O)cccc(Cl)c1 32039,C1(C(=O)NC(C(C)C)(C)CNC(=O)Cc2cnsc2)CCc2nncn2CC1 32040,C1(C(=O)NCCSCCC=C)C(CNC(=O)CN2CCCC2)C1(C)C 32041,CC1CN(C(c2cnncc2O)=O)CC1(C)CNC(=O)C1=CCCC1 32042,c1(CC(=O)NCCC(=O)NCCC(C)C)ccc(F)cc1F 32043,C(=O)(CCC(=O)c1cccnc1)NCCOC1CCN(C(C2C(OC)C2)=O)C1 32044,N1(C(C(C)NC(C)(C)C)=O)CCN(C(c2cccnc2)=O)C(CC(F)(F)F)C1 32045,N1(C(c2ncc(C)cn2)=O)CC2CCC1C(CNC(c1ccc(F)c(Cl)c1)=O)C2 32046,N1(C(CC(C)OC)=O)CC2(C1)CN(C(C1CCn3nncc3C1)=O)CCO2 32047,C(=O)(C(C)CC(C)C)NCC(CNC(c1cccc(C(=O)OC)n1)=O)(C)O 32048,CN1C(=O)CC(N2CC(CNC(=O)NCCS(C)(=O)=O)C2)C1=O 32049,c1(C(N2CC(O)CC(NC(=O)C(F)F)C2)=O)ccc2c(c1)CCO2 32050,C=CCCCCCC(=O)N1CCCC1(C(=O)NCC1CN2CCC1C2)COC 32051,c1(CC)ccc(S(C)(=O)=O)cc1C(N1CCOC(COc2ccccc2)C1)=O 32052,c1(CN2C(CC(=O)Nc3cc(C(=O)OC)sc3C)CCC2)c(OC)cccc1Br 32053,C(=O)(CCCCC(F)(F)F)NCCC1(C)CCN(C(=O)Cc2cc[nH]n2)C1 32054,N1(C(CCC(C)(F)F)=O)Cc2ccccc2CC1CNC(=O)CCOC1CCC1 32055,c1(CC)ccc(Cl)cc1NC(C1CCCN(Cc2cccnc2C(=O)O)C1)=O 32056,c1(NC(c2ccccc2)CNC(N)=O)ncccc1S(=O)(=O)NC1CNC1 32057,Cc1ccn(CC(C)(O)C(=O)NC2CC(NC(=O)C(C)(C)N3CCC3)C2)c(=O)c1 32058,CC1CCc2[nH]nc(C(=O)NC34CCCC3CN(C(=O)CCCC(N)=O)C4)c2C1 32059,N1(C(c2c(CC)c[nH]n2)=O)CC=CC(NC(=O)COC)C1 32060,Cc1nccc(C(=O)N(C2CN(C(=O)CC3CCNC(=O)C3)CC2(C)C)C)c1C 32061,C1(NC(Cc2ccc(OC)nc2)=O)CC2(C1)CC(NC(c1noc(C)n1)(C)C)C2 32062,c1(OC)ccc(F)c(F)c1CN1CCOC(C(=O)Nc2ccc(C#N)cc2O)C1 32063,C1(C(N2CCCC(CNc3ncc([N+](=O)[O-])cn3)CC2)=O)CCC2CCCCN12 32064,c1(C(N2C(C(=O)NCCOc3ccc(C)cc3)CC(=C)C2)=O)ccc(C#N)cc1 32065,Cc1cc(C(=O)NCCC(C)CCNC(C2(C(F)(F)F)CC2)=O)nn1C(C)(C)C 32066,C(c1ccncc1)=C(C)C(=O)OCC(=O)NCC(C1CCCCC1C)=O 32067,c1(C(N2CCCC(NC(c3ccc(C#C)cn3)=O)C2)=O)ncnc2c1ccn2C 32068,C1(CNC(c2c(CC=C)cccc2)=O)CCN(C(C2CC(F)CN2C)=O)C12CC2 32069,N1(C(c2c(C)ocn2)=O)CC2C(CN(C(=O)CC3CC4CC4C3)C)C2C1 32070,CC1CN(C(C2CC3CC(=O)C2O3)=O)CC1(C)C(N1CCC(C)(O)C1)=O 32071,Cc1csc2nc(CC(N3CC(NC(C4(C(N)=O)CC4)=O)CCC3C)=O)cn12 32072,C1(C(=O)NC2CC(CNC(C(c3ccncc3)C)=O)C2)COCCN1C 32073,c1(OC)ccc2nc(CNCC3(F)CCCC3)ccc2c1 32074,N1(C(Cn2c(C)nnn2)=O)CC(NC(c2cc(O)nc(Cl)c2)=O)CC(F)C1 32075,c1(C(CCO)N(CC(COCC)COC)C=O)ccc(OC)cc1 32076,C1(C(=O)NCC2(C)CN(C(=O)Cc3ccc(F)cc3)C2)C2CCC(F)C12 32077,c1(C(=O)NCC(CCCC)NC(c2occc2Cl)=O)cc(N(C)C)ccc1F 32078,C(=O)(C1=CC2C=CC1C2)N(CCCCCNC(=O)CCC1CCCOC1)C 32079,N1(C(c2ccc(C(N)=O)o2)=O)CC2(CC(NC(=O)CCc3csnn3)C2)C1 32080,C12(C(=O)NCc3ccc(C)cc3C)C3CCC(CC13)C2(F)F 32081,c1(C(=O)NCCCC(C)NC(c2c(OC)noc2C)=O)ccc2ncsc2c1 32082,c1(SCC)ccc(NC(=O)NCC2(OCC)CCOC2)o1 32083,C1(C)(CC)C=C(C(=O)N2CC3CC3(C(N3CCC(C(=O)OC)C3C)=O)C2)C1 32084,C(CCC(C)C)(C(=O)NOCC(O)CO)NC(C(CC=C)C(C)C)=O 32085,C1(CC)CC(C(=O)N(C2CCCC(O)C2)C)CCN1C(=O)C(F)C(F)(F)F 32086,CCCCCS(=O)(=O)CC(=O)NCC(C)NC(=O)C#CC1CCCCC1 32087,c1(C(=O)NCC(CC)NC(c2cnn(CCO)c2C)=O)ncc[nH]c1=O 32088,C1(NC(C(CC)(F)F)=O)COC2(C1)CN(C(=O)Cc1c(F)cccc1C#N)C2 32089,C(=O)(C(CNC(=O)CC1CSC1)CC(C)C)NC(C#C)(C)C1CCC1 32090,CC1(CCNC(=O)CC2CCC(=O)O2)CCN(C(c2cnoc2C2CCC2)=O)C1 32091,N1(C(c2nc(OC)c(C)s2)C(=O)NC2CC2)CCCC2CCC(C)CC12 32092,C(C(CC(F)(F)F)NC(c1cnc(O)o1)=O)NC(CCC1CCC(=O)NC1)=O 32093,N1(C(CCN(C(c2ccoc2C(F)(F)F)=O)CC)=O)CCCC(CN(C)C)C1 32094,c1(CC)c(C(=O)NCCC2(NC(c3cc(N)ccc3C)=O)CC2)cccc1C 32095,N1(CC(=O)NC2(CCC(N3CC4(CCC4)C3)=O)CCC2)CCCCC1=O 32096,c1(C(=O)NCC2(NC(c3c(CC)nccc3)=O)CC2)cc(O)ccc1C 32097,N1(C(C2=C(C)CCC2)=O)CC(NC(=O)C(C)OCCC(C)C)C(C2CC2)C1 32098,c1(COC(=O)NC(c2c(C)sc(Br)n2)C(=O)OC(C)(C)C)cc(F)c(O)c(F)c1 32099,c1(C(=O)NCC(C)C#N)cnc(CNC(C2CC2(Cl)Cl)=O)nc1 32100,c1(C(=O)NCCOCCC#C)ccc(Br)cc1SC 32101,CC1(C)OCCOC1C(=O)NCCC1CCN(C(=O)CN(C2CCCC2)C)CC1 32102,CCC(C)(C)CCCC(=O)NC1C(C)CN(C(c2cnn(CCF)c2)=O)CC1C 32103,CCS(=O)(=O)CC(=O)N1CCN(C(c2cc(OCC)cc(=O)o2)=O)CC1CCO 32104,C(CN=S(C)(C)=O)N(C)C(c1csc(C(=O)OC(C)(C)C)n1)=O 32105,CN1CCC(C2(C(N3CC(CNC(c4ccc(Cl)o4)=O)C3)=O)CC2)CC1 32106,C1(C(N2C(CC(=O)OC)CCC2)=O)CCCN(C(C2CC2(Cl)Cl)=O)C1C 32107,C#Cc1cccc(C(N2CCSCC2C(=O)N(C)C(C)C2CC2)=O)c1 32108,C(=O)(C1=C(C)NC2=NCCCC2=C1)NCC1N(C(COCCCCC)=O)CC1 32109,CCC(CNC(C1CC(=O)N(c2cccc(F)c2)C1)=O)N=c1[nH]nc(C2CC2)s1 32110,N1(C(C2CN(C(C3N(C)C(=O)CC3)=O)CC(F)C2)=O)CCN2CCOCC2C1 32111,c1(CC(=O)N(C2CN(C(c3nonc3N)=O)CC2F)C)cncnc1O 32112,C(=O)(CC(O)CC1CC1)NC(CNC(CCSCCC)=O)C(C)C 32113,c1(CC)ccc(C(=O)NC2CN(C(=O)CSC(F)(F)F)CC2C(F)F)cn1 32114,c1(N2CCC(C)(CNC(C)CCO)CC2)ccc(S(=O)(=O)N2CCCC2)cc1Br 32115,C1(NC(=O)C(CC2CC2)NC(C23CC2CNC3=O)=O)C2CCCCCC12 32116,c1(C(=O)NC(CNC(C(C)=CC)=O)(C)C2CC2)cc(C)c(-c2ccc(Cl)cc2)s1 32117,C1(CC#C)(C(=O)N(C(=O)CCC=C=C)CCCCC)CCCCO1 32118,n1(CCS(C)(=O)=O)ccc(=NC(=O)C2COC(C)(C)C2)[nH]1 32119,c1(C(=O)NCC(C)N(C)C(C(C)C(N2CCCCC2)=O)=O)[nH]ccc1C1CC1 32120,c1(C(C(=O)NCCCCNC(C(SC)SC)=O)F)ccccc1 32121,CC(=O)CCCC(C)C(=O)N1CC(C)CC1C(N1CCC(OCCF)C1)=O 32122,C(=O)(C(C(C)C)n1cncn1)N(CC(CNC(C(CC)n1cncn1)=O)(C)C)C 32123,C(=O)(C(O)CC(F)F)NC(CCNC(CCc1cnc(C)o1)=O)C 32124,c1(C(=O)NC(c2ccc(Cl)cc2)C(C)C)ccc(F)c(-c2cc(F)nc(F)c2)n1 32125,C1(CNC(N2CCN(Cc3ccccc3)CC2)=O)CCCCC(F)(F)C1 32126,N1(C(c2cc(CCC)[nH]n2)=O)CCC(C)C(NC(c2ncc(N(C)C)cn2)=O)C1 32127,C1(O)(CC(=O)NC2C(OC3CC3)CN(C(CN(C(=O)OC)C)=O)C2)COC(C)(C)C1 32128,C1(C(=O)NC2CCN(c3ccc([N+](=O)[O-])cc3)C2)CCCC2(C1)CC2(F)F 32129,CCCCC(O)C(=O)NCCC(C)NC(=O)C(=O)NCC(F)(F)F 32130,C(C(C)(C)CNC(C1(Cl)CC1(F)F)=O)N(C(=O)CCCc1cccs1)C 32131,c1(C(N2CC(C)(NC(C(C=C=C)C)=O)C2)=O)ccc(C(=O)N(C)C)nc1C 32132,c1(C(C)NC(=O)NCC(C)(C)C(F)F)ccc(-c2ccccc2)c(F)c1 32133,C(C)(CCCNC(=O)C(F)(F)c1nccs1)NC(C(C)NC(C)=O)=O 32134,C12(C(=O)NC(CCCCC)C)CCC(CN(C(c3n[nH]c(C)c3O)=O)C1)C2 32135,Cc1c(C=CC(=O)N(C)CC2CCCN2C(C2CCOCC2)=O)cnn1C 32136,Nc1ccc(-c2cn(C3CC(NC(c4nc(Cl)cs4)=O)C3)nn2)nc1 32137,C1(CNC(c2coc(O)n2)=O)CC(O)CN1C(=O)Cc1ccsn1 32138,C(=O)(CCC(=O)NC(C)CN(C(=O)CC1(O)CCC1)C)N(CC)CC 32139,CCC(CC)N=c1[nH]c(=NCC2CCCC2OC)[nH]c2cc[nH]c12 32140,c1(OCCC)c(Cl)cc(NC(c2cnc(OC)c(F)c2)=O)cc1Cl 32141,Cc1c(OC(C)C)cccc1N=c1cc(N)nc(C(C)C)[nH]1 32142,CC(C)S(=O)(=O)CC(=O)NCC1(CNC(C2CCCO2)=O)CCC1 32143,c1(C(=O)NCCCC(C)NC(=O)C(C)C#N)cncc(C(=O)OC(C)(C)C)c1 32144,C1(CNC(CCCC=C)=O)CC2CCC1N(C(=O)Cc1cc(C)cs1)C2 32145,C1(CNC(C2CC=C(C)CC2)=O)(CO)CCN(C(c2nn(C)cc2Cl)=O)CC1 32146,C1(SCC(=O)NCC(CC)NC(c2cn(C3CC3)cn2)=O)CCOC1=O 32147,c1(CN2CCC(NC(c3cc(Cl)ccc3Cl)=O)C(O)C2)cncc2ccccc12 32148,C1(NC(C(CC(C)C)N(C)C)=O)COC2(C1)CN(C(=O)Cc1ccncc1Cl)C2 32149,CC1(C)CC(C(=O)NCC(O)CC2CCC2)N(C(=O)C=Cc2ccco2)C1 32150,C1(CCNC(=O)Cn2cccc2)CCCN(C(c2sc(Cl)cc2Cl)=O)C1 32151,c1(C(N2CC(CC(C#C)C)C2)=O)cc(F)c(C)cc1Cl 32152,N(C1CCc2ccccc21)C(C12CC(Nc3nccc(Br)n3)(C1)C2)=O 32153,C1(C(=O)NCC2CCCS2)CCC(NCCCN2CCC2)CC1 32154,C(=O)(C(F)(F)C(C)O)NC(CN(C(c1c(C(=O)OC)nn(C)n1)=O)C)C 32155,Cc1cn2cc(NC3(CO)CCN(C(=O)Nc4ncccc4Cl)C3)ccc2n1 32156,c1(C(=O)NC23C(CN(C(C(C=C)(C)CC)=O)C2)C3)ccc([N+](=O)[O-])c(N)n1 32157,N1(C(c2ccc(C)cc2)=O)CCCN(C(=O)C(CO)c2ccccc2)C(CO)C1 32158,C1(COC)CN(C(=O)C=C(C)C(C)(C)C)CCN1C(C1CCC12CCC2)=O 32159,C1(C(N2CC(=C)C2)=O)CC(=O)CN1C(=O)CCc1cccn1C 32160,C1(NC(CC(CCC)(C)C)=O)CC(C2CCN(C(=O)C(C)c3ccco3)CC2)C1 32161,C1(N(C(CN(C)CC)=O)C)CCC2CN(C(c3ocnc3C3CC3)=O)CC12 32162,C(CC(=O)NCC(CO)NC(=O)CC1CC(OC)C1)OCC#C 32163,Cc1csc2c(CC(N3CC(C4(NC(=O)C(C)CN(C)C)CC4)C3)=O)cccc12 32164,CCC(C(=O)N1CC2(CC2)CC1CNC(c1cn(CCCF)nn1)=O)C(C)C 32165,c1(C(N(CC(C)CNC(=O)CCn2cnccc2=O)C)=O)ccc(N)c(Cl)c1O 32166,CCC(C)CCCC(=O)N1CC(NC(C2CN3CCC2CC3)=O)C(C)C1 32167,Cc1c(C(=O)NC(C)C(CO)NC(=O)C2=NOC(C)(C)C2)nc2sccn12 32168,c1(SCC)ccc([N+](=O)[O-])cc1C(=O)NC1CN(C(=O)C#CC2(C)CC2)CC1O 32169,CC1(C)c2[nH]nc(NC(c3ccc(Cl)c(Cl)c3Cl)=O)c2CN1C(=O)C=CC1CC1 32170,C1(c2ccccc2)(C(=O)NCC2CCN2C(=O)COc2ccccn2)CCCO1 32171,c1(C(=O)NCC(CC)NC(c2cnccn2)=O)nonc1N 32172,Cc1nc2c([nH]1)CC(C(=O)N(C)CCNC(c1ccc(C(C)C)o1)=O)CC2 32173,Cc1ncc(C(N2CCCC2CC(=O)NCc2cnn(C(C)C)c2)=O)c(=N)[nH]1 32174,Cc1ccc(CC(=O)NC(C)CNC(C2CCCC(C)O2)=O)c(Br)c1 32175,Cc1cc(N2CCC(NC(C3CCCC3(C)C)=O)C(F)C2)nc(S(C)(=O)=O)n1 32176,c1(C(=O)NC2CC(CNC(C(C)(O)C3CCC3)=O)C2)cc(Cl)nc(Cl)c1 32177,C=C(C)CC(C(=O)NC1CN(C(C2CC(C)(C)CN2C)=O)C1)OC 32178,c1(C(=O)NCC2CCCN(C(C(C)(C)CC#N)=O)C2)cc(F)cc2nc[nH]c12 32179,C(=O)(C1CCCc2cncn21)NCCCCNC(C(C)N(CC(F)(F)F)C)=O 32180,Cc1nc(C(N2CCC(C(=O)NC(C(=O)OC)C3CC3)C2C)=O)c(C)s1 32181,c1(C(=O)NCC(C2CCC2)NC(C2CC2c2ccsc2)=O)c[nH]nc1C(F)F 32182,C1(NC(C)=O)CCCC(NC(c2cc(-c3ccccc3)[nH]n2)=O)CC1 32183,N1(C(C(C=C)O)=O)CC(C(N2C(C(=O)OC)CC2C)=O)CC(C)C1 32184,Cc1coc(C(=O)NC(C)(C)C(C)NC(c2cc(C(C)C)no2)=O)c1C 32185,C1(C(=O)NCC2N(C(C(c3cccc(Cl)c3)CC)=O)CCC2)CCC2CC2C1 32186,C1(OC(=O)NCCC(=O)N(CCC)CCC)CC2=NC=CN1C2 32187,CCCCCCCCCCC(=O)NC(C)CN(C(=O)C(c1ccc(Cl)cc1)O)C 32188,c1(C(NC(=NC2CC2)NC2CCC3(CC3)C2)C)cc2cccc(F)c2o1.c1(OC)nnn[nH]1 32189,c1(C(N2CC(N(C(C=CC(C)C)=O)C)C(F)C2)=O)cc2nccn2c(O)n1 32190,C1(CNC(CCC(C)C)=O)CC2CCC(C1)N2C(=O)NC1(c2cccnc2)CC1 32191,c1(C(C(=O)NC2(C=C)CNC2)(F)F)ccccc1Br 32192,c1(C(N2C(C#C)CCC2)C(=O)NC2CC(F)(F)C2)cccc2[nH]ncc12 32193,c1(C(N2CC(SC)C(NC(=O)C(C(C)C)N(C)C)C2)=O)cnn2ccn(C)c12 32194,CC1(CNC(c2[nH]ccc2CNC(C2OC3CCC2C3)=O)=O)CCCCO1 32195,CCCCC(CNC(C1CC(OC)(OC)C1)=O)NC(=O)CC1CCC(=O)N1C 32196,C1(CNC(=O)CCC2CCC(=O)N2)CN(C(C2CC2F)=O)CCC12CCC2 32197,c1(C(=O)NCC(C)N(C(C)=O)CC)cncc(N)c1.C1(=O)C(C(C)C)N1 32198,c1(CC(=O)NC(CNC(C(C)SC2CC2)=O)CO)cccc2cn[nH]c12 32199,CC1(C)C(C(=O)NCC(P(C)(C)=O)c2ccccc2)(CO)C1(C)C 32200,C(=O)(C(F)(F)CC(C)C)NC(CNC(c1c(C)nc(CO)s1)=O)CO 32201,C1(CNC(CC(C)C2CCCO2)=O)CCN(C(=O)C(C)(C)n2ccnn2)CC1 32202,c1(C(N2CC(SC)C(NC(=O)CCSC(F)(F)F)C2)=O)ncnc2c1ccn2C 32203,c1(-c2cc(C)cc(OC)c2F)cccc2[nH]nc(C(=O)Nc3conc3C)c12 32204,Cn1ccc(S(=O)(=O)NC2(CNCc3cnc(Cl)cc3F)COC2)n1 32205,C#CCCCC(C)C(=O)N(C1CC(C#N)C1)CC(=O)NCC1CCC(=O)NC1 32206,N1(C(C2C3CN(C)CC32)=O)CCC2C(CCN2C(c2ccc(F)cc2Cl)=O)C1 32207,C1(NC(C(C)OC)=O)CCN(C(c2cnc(-c3ccccn3)nc2)=O)CC1O 32208,N1(C(C(c2n(C)cnc2)O)=O)CCN(C(c2cocn2)=O)C(CO)C1 32209,c1(OC)cc(C)cc(C(=O)NCC2CC(OC)CN2C(=O)CC(F)F)c1C 32210,c1(C(=O)NC2CC3(CC(CNC(C(CC#C)(C)C)=O)C3)C2)cc(C)c(C)nc1C 32211,c1(C(N2CC(CC(=O)NOCC(C)C)(OC)C2)=O)sc(O)nc1C 32212,c1(OC)nccc(C(=O)NC23CC(CNC(=O)C(CCSC)NC(N)=O)(C2)C3)n1 32213,C1(C(=O)NCCNC(C2(C(=O)OC(C)(C)C)CC2)=O)CC2(C1)C(F)(F)C21CCC1 32214,Cc1c(CN(C)C(=O)NCCC2COCCO2)cccc1F 32215,N1(C(C(CNC(=O)COC2CCOCC2)O)=O)CCC2(CC1)CSC2 32216,C12(NC3CCN(c4ccccc4)C3)CC(CO)C(CO1)C2 32217,c1(CC)nc(CNC(=O)C(F)NC(C2CC2C(C)OC(C)(C)C)=O)n[nH]1 32218,C1(NC(CNC(C(CC)CC)=O)=O)CC2CC(NC(C3CNC(=O)C3)=O)CC2C1 32219,C1(CNC(c2ccc(OC)cn2)=O)(OC)CCN(C(C2CCCS2)=O)CC1 32220,Cc1nc(N(C)CCN(C)C)cc(N2CCOC(Cn3ccnc3C)C2)n1 32221,C(=O)(C1=C(C(=O)OC)C(c2ccc3cnccn23)NC(=O)N1C1CC1)OC 32222,N1(C(C2CCCC(C(=O)OC)C2)=O)CC2(CCCCN(C(c3ccsc3)=O)C2)C1 32223,c1(C)sc(C)c(Br)c1C.c1(C(COC)NCC=C)nnnn1Cc1nnn(C)n1 32224,c1(OC)cnc(NC(C2CC23CN(Cc2cc(C)[nH]n2)C3)=O)c(F)c1 32225,N1(C(C2(COC)CCOCC2)=O)CCN(C(=O)C(C)n2ccnc2)CC12CC2 32226,C(=O)(C1=NOC2COCC12)N1C2C(C(N3CC4CC4(CO)C3)=O)C(C2)C1 32227,C(CC(=O)N1CCN(C2CCC2)CC1)(C(C)OC)NC(C(COC)COC)=O 32228,N1(C(c2csc(C3CCCCC3)n2)=O)CCC(O)C(NC(C2(C3CC3)CC2)=O)C1 32229,CC(CC(N)=O)C(=O)NCC(C)(C)CC(=O)NCC12CC(CCO1)C2 32230,Cc1cc(F)sc1C(=O)NC1(c2ccccc2)CCN(C(C2CNC(=O)C2)=O)C1 32231,N1(C(C(C)CN(C(=O)CCC2CCC(=O)C2)C)=O)Cc2ccnn2CC1C 32232,Cc1ccc(N(CCCNC(=O)C2=CC3CCCC23)C(C)C)c([N+](=O)[O-])c1 32233,CN1CCC(C)(C(=O)NCCC2(CNC(=O)C(F)CC3CCCCC3)CC2)C1 32234,C=C(C)CC(C(=O)NC(C(=O)NC)C1CC1)NC(C1(C)CCC(C)C1)=O 32235,c1(CC(N2CC(O)(CN(C)C(c3cccc(F)c3O)=O)C2)=O)cc(Cl)ccc1Cl 32236,CC1CN(c2nc(C3CCOCC3)ns2)CCC1NC(c1ccnc(O)c1)=O 32237,c1(C(=O)NC(C2CCN(C(C3C(CC)C3)=O)C2)C)ccc(Cl)nc1 32238,C1(C(=O)NCC2C(C)(C)C(NC(c3ccc(Cl)[nH]3)=O)C2)CCc2[nH]nc(O)c2C1 32239,C1(CNC(C(C)OCC(C)C)=O)CCCCN(C(=O)C(O)c2ccco2)C1 32240,N1(C(C2N(C)CCOC2)=O)CC2(CCN(C(C34COC(C3)C4)=O)CC2)C1 32241,CCC(C(=O)NCC(COC)NC(c1cccc(C)c1F)=O)C(C)(F)F 32242,C1(C(=O)NCC(C)NC(=O)CC2(CO)CC2)CC2C(C1)C2(C)C.C(C)(C)(C)OC(=O)N 32243,C1(NC(CN(CCOC)C)=O)CN(C(=O)C(c2ccc(Cl)cc2)C)CC12CC2 32244,N1(C(=O)Cc2cn[nH]c2)CCCC(C2CN(C(C3COCCC3(F)F)=O)C2)C1 32245,C(CC(C)C)(C(=O)N1CCC(O)(CO)C1)NC(CN(C(C(C)C)=O)C)=O 32246,c1(C(N2C(C)CC(NC(C3CCCC3(C)C)=O)CC2)=O)cncc(N=[N+]=[N-])c1 32247,N1(C(CNS(NC)(=O)=O)=O)C2CCC1CN(C(=O)COc1ccc(N)cc1)CC2 32248,C(=O)(N=c1[nH]nc(Br)s1)NCC1CCCN(C(c2ccsc2)C)C1 32249,C1(CCNC(CCN(C)CC)=O)CCCCN1C(c1ocnc1C1CC1)=O 32250,c1(C(=O)NC2C(NC(CC3OCC(C)(C)OC3)=O)C2)ccc(Cl)c(Cl)c1O 32251,c1(C(N2CCCC(N(C(c3cnco3)=O)CC)C2)=O)cnn2cccc(Cl)c12 32252,c1(C(=O)NC2(CNC(c3cnc(C)[nH]3)=O)CCCCC2C)cn2cnnc2cn1 32253,n1(CCC)cc(Cl)c(C(=O)NCC2(OC)CCN(C(=O)Cc3cnn(C)c3)C2)n1 32254,C#CC1CC1C(=O)NC1CC(N(C(=O)CC2CCN2C(=O)OC(C)(C)C)C)C1 32255,N1(C(c2c(C)nsc2)=O)CC2(CC(C(=O)NCC(C)(O)C3(C)CC3)CO2)C1 32256,c1(C(N2CCN(C(CCN(CC)CC)=O)CC2C(F)F)=O)nc(O)nc(O)c1F 32257,CC(C)(C)CC(F)C(=O)N1CC(CNC(=O)CSCC(N)=O)C(F)(F)C1 32258,CC1(CCC(N2CCOCC2)=O)CN(CC(C(=O)CCC2CCC(=O)C2)=O)C1.N 32259,Cc1cc(C(C)C)ccc1C(=O)NC1C2CC1N(C(c1cncnc1C)=O)C2 32260,N1(C(c2cc(C(C)C)on2)C(=O)NCC(=C)C)CCC2CC12C(=O)OOCC 32261,c1(CC(=O)NC2CC(NC(c3ccnnc3O)=O)C2)cc(F)cc(F)c1Br 32262,N1(C(CC(C=C)C)=O)C(C)CC2CN(C(=O)C(C3(O)CCCC3)F)CC12 32263,C(C(F)(F)CCC(=O)NC(CO)CC(C)(C)C)n1cc(-c2cc(C)[nH]n2)nn1 32264,Cc1c(S(N)(=O)=O)cnc(NCCC(c2ccc(Br)cc2)O)c1Br 32265,c1(C(N2CC3C(NC(c4ncn(C)c4)=O)(C3)C2)=O)c(F)cc(F)cc1Cl 32266,c1(C(=O)NCC(C)CNC(C2(N(C)C)CC2)=O)cccc2cnccc12 32267,C1(C(=O)NC(C#C)C2CC2)C2CC3C(C2NC(=O)CCCCSC)C13 32268,c1(CC(C(=O)OC)Nn2cc(C3CC=CCC3)nn2)ccc(OC(F)(F)F)cc1 32269,c1(CN2CC(NC(c3c(C)ccc(Br)c3)=O)C(C#N)C2)ccc2nc[nH]c2c1 32270,C(C(=O)Nc1cncnc1C)(C(C)(C)C)NC(CCSCCCC)=O 32271,N1(C(COc2cccc(OC)c2)=O)CC2CC(NC(=O)C(C#N)C(C)C)C(C2)C1 32272,c1(C(N(CC(CC)NC(c2c(CC)cc[nH]2)=O)C)=O)nccc2ccn(C)c12 32273,C1(NC(C=C(C)C)=O)CN(C(c2snnc2C(C)C)=O)CC1C 32274,C1(CC)CN(C(C2C(C)C2C)=O)CC1C(=O)N(C)CCOC(C)=O 32275,N1(C(C(CCCC)O)=O)CCN(C(C2CC(OC)C2)=O)C2(CCC2)C1 32276,C1(C)(C(=O)NCC(=C2CN(C(CCCOC(C)C)=O)C2)F)CCCS1(=O)=O 32277,C1(C(=O)NC2(C)CC(NC(=O)CC3CC3(Cl)Cl)C2)COCCN1CC(F)F 32278,c1(NC(C(N2CCC(N(C(c3cnccc3C)=O)CC)C2)C)=O)cnc(C)nc1 32279,CC1CC2CC1CN(C(c1cc(F)ccc1F)c1ccccc1)C2 32280,N1(C(C2OCCN(C(C)=O)C2)=O)CC2(CCN2C(=O)C2=CCOCC2)C1 32281,C1(C(=O)NC2CCC(CNC(C(C)C#N)=O)C2)CC2(CC(=O)N2)C1 32282,O=C1C=C2CN(C(=O)CC3CN(C(c4n[nH]cc4I)=O)CCO3)CCC2S1 32283,C1(CCNC(=O)CCCN2CCCC2)CC(F)(F)CN1C(=O)Cn1cnnc1 32284,c1(C(=O)NC2(C)CC(NC(c3scnc3C(C)(C)C)=O)C2)ccncc1O 32285,C(c1cnc2ccccc2n1)=CC(N1CCC(NC(C=C(C)C)=O)C(C)C1)=O 32286,S(=O)(=O)(c1ccc(NC2CCOC(C(C)C)C2)cc1Br)NCC(C)(C)OC(C)C 32287,c1(C(=O)NCC(C)(CC(C)C)NC(C(CC(=C)C)C)=O)cn2cc(C)ccc2n1 32288,C1(CCNC(C2C(OC)CC2)=O)CCCCN1C(c1cccnn1)=O 32289,c1(NC(c2c(OC)n[nH]c2)=O)ccc(-c2ccccc2)c(F)c1 32290,C1(CNC(CC=C(C)C)=O)CC2(CCN(C(c3cn(C(C)C)cc3C)=O)C2)CO1 32291,CCC(C(C)(C)O)NC(c1cnn(CCNC(C2CCC(=O)C2)=O)c1)=O 32292,C(=O)(CCCCC(N)=O)NC(C(=O)NC1CCCN(C)C1)CO 32293,C(N=c1[nH]c(=NCCN(C)C(C)C)[nH]c2cc[nH]c12)C1N(CC)CCCC1 32294,C#Cc1ccnc(C(N2CCN(C(=O)C(CC)CC=C)C(C(C)(C)C)C2)=O)c1 32295,C1(F)(CNC(C(CCCC)C)=O)CCCN(C(=O)Cc2ccc3occc3c2)CC1 32296,CC1(C)CC(CNC(=O)C(F)=C2CCC2)N(C(=O)CC2CC3CC3C2)C1 32297,C(=O)(CCC(C)S(C)(=O)=O)NC(CNC(c1c(C)nn(C2CC2)c1Cl)=O)C1CC1 32298,CCC(C)C(C(=O)N1CCOC2CC12)N(C)C(C1CCN(CC)CC1)=O 32299,c1(CC(N2C(C)C(NC(=O)CCn3cccn3)CC2)=O)cccc2sccc12 32300,CC(c1ccccc1Cl)=CC(=O)NC1CC(NC(c2cc(C)c(C#N)cn2)=O)C1 32301,Cc1ccc(O)c(C(=O)NCCCNC(c2ccn(C)n2)=O)n1 32302,c1(C(N(C2CC3CNC2C3)C(C(C)C)CO)=O)ccc2cnccc2c1 32303,N1(CC)CCCC(NC(C23CC2CCN3C(=O)C(C)c2cc[nH]n2)=O)C1 32304,c1(C(C(=O)NCCCNC(C)=O)N(CC=C)CC#N)nn(CC)nc1C 32305,N1(C(c2ccc(CCC)[nH]2)=O)CC(NC(c2cccc(N)c2)=O)CC1(C)COC 32306,C1(C(=O)OC)C2CC1N(C(=O)C(C1CCN(C(=O)C(C)(C)Cl)C1)F)C2 32307,c1(NCC(CC)CO)nc(N2CC(CO)C(C)C2)nc2c1ncn2C(C)C 32308,N1(CC)CC(C(=O)N(C)CCNC(c2ccnc(OC3CCC3)c2)=O)NC1=O 32309,C(CCCCCC(=O)NC1CC(CC(=O)OC)C1)n1cc(-c2c(C)ncs2)nn1 32310,N1(C(COC)=O)CCCC2(NC(c3ncc(C(F)(F)F)s3)=O)CC2C1 32311,C(CC(=O)NOCCC(C)O)(C(F)(F)F)NC(C1(COCC)CC1)=O 32312,c1(C(N2CCC(C)(NC(c3nc(C)c(C)[nH]3)=O)CC2)=O)cnc(O)c2ccsc12 32313,C(CC(C(=O)NCCc1nccn1C)NC(=O)CCc1ccc(C)o1)=CC 32314,c1(C(=O)NCC2=CCN(C(C3CC=CC(O)C3)=O)CC2)cccc2ccoc12 32315,C(CNC(c1cc(OC)cs1)=O)(CCC)NC(C(C)=C(CC)C)=O 32316,C12(C(N(CCN(C)C(C3(n4ccnn4)CC3)=O)C)=O)CC(C1)C(C)(C)O2 32317,C1(F)(C(=O)NCC2CC(NC(CSc3n(C(C)(C)C)cnn3)=O)C2)CCCCC1 32318,N1(N(C(C(C)C)=O)C)CC2(CCOCC2)C1.N12CC(CC1C)OC2=O 32319,O=S(=O)(c1ccc(NCCCCCF)c(Br)c1)NC1C=CCCCC1 32320,N1(C(C2CC(=O)N2)=O)CCC(C2CCCN(C(c3ccn(O)c(=O)c3)=O)C2)C1 32321,Cc1cnc(N2CC3(CCCC3NC(c3ccc(Cl)cc3C)=O)C2)c([N+](=O)[O-])c1 32322,C(=O)(CCCCCF)NC1CC(C)(NC(C2CCCC(C(F)(F)F)C2)=O)C1 32323,C1(C(=O)C)CCCN1NC(=O)C=Cc1cocn1 32324,N1(C(c2cc(CCC)[nH]n2)=O)CCCC(N2CCN(C(C3CCOC3)=O)CC2)C1 32325,Cc1ccnc(C(C)(C)C(=O)NC(C)CN(C(=O)C(F)OC(F)(F)F)C)c1 32326,N1(C(c2c(C)c(F)ccc2)=O)CCCC2CN(C(=O)C3=CCCCC3)CCCC12 32327,C#CCCCCC(=O)NC1CC1CNC(c1ccc[n+]([O-])c1)=O 32328,c1(CN(C(=O)C=CC2CC2)C)cccc(O)c1 32329,N1(C(C(OCC)OCC)=O)CCC(C(=O)NC2CCC2C(F)(F)F)C(O)C1 32330,C(=O)(CCC(C)(C)N(C)C)NC(CC)CC(=O)NCC1CCC(C2CC2)O1 32331,C1(CN(CC)CCN2CCCC2=O)CCCN1N(C)C 32332,c1(C(N2C(C)CC(NC(=O)COc3ccsc3)C2)=O)cc(F)cc2nc[nH]c12 32333,CN1CCCC1C=CC(=O)NCC1(O)CCN(C(c2cscn2)=O)C1 32334,c1(CN2C(C)(C(=O)Nc3cccc4c[nH]nc34)CC2)ccc2c(c1)CCCC2 32335,C1(C(N(C2CN(C)C2)C)=O)CC12CCN(C(c1cscc1Cl)=O)CC2 32336,C1(CS(C)(=O)=O)CN(C(=O)CC2(O)CCC2)CCN1C(c1cc(F)c[nH]1)=O 32337,N1(C(C(Cn2ccnn2)NC(CCCOC)=O)=O)CC2C(C1)C2(C)C 32338,c1(C(N2CCC(C)(NC(c3[nH]cc(C)c3)=O)C2)=O)cc(C)nc2c(Br)cnn12 32339,N1(C(C(C)=CC)=O)CC(C2CN(C(c3cc4ncccc4s3)=O)C2)C1 32340,C12(C(N(CC)CC3CCOC3)=O)CC1CN(C(=O)C(C)=NOCC#N)C2 32341,c1(C(N2CCC(N(C(=O)C(F)C(F)(F)F)CC#C)CC2)=O)cc(C)nc(Cl)c1N 32342,C1(CC#C)CCCCN1C(=O)C(C)N(C)C(c1ncccc1F)=O 32343,C1(C)(C(N(C2CC(C#N)C2)CC(=O)NCCCC2(C)CC2)=O)CCOC1 32344,C(C(O)C(=O)NC1CCC1NC(=O)COCCSC)=CC 32345,Clc1ccc(CN2CCC2COc2ccccc2)cc1Cl 32346,C(CC(=O)NOCC(=O)N(C)C)C1CC(NC(C2C(C)C2)=O)C1 32347,C1(O)(CNC(CCc2onc(CC)n2)=O)CCN(C(c2snnc2C2CC2)=O)C1 32348,N1(C(C(C(=C)Cl)(C)C)=O)C2CCCC1CN(C(C1COCCC1C)=O)C2 32349,CCCCC(C)C(=O)N1CCN(C(c2ccnn2C(C)C)=O)C(C(C)(C)C)C1 32350,N1(C(C(C)(C)NC(C)=O)=O)CC2(C(=O)NCC(F)Cl)CC1CO2 32351,c1(SC)nc(N2CCC(NC(c3ccn(C)c3)=O)C(F)C2)cc(C(F)F)n1 32352,C(=O)(C1=COCCC1)N(C)CC1CCN(C(c2c(C)n[nH]c2)=O)C1 32353,N1(C(CN(C)C(C2CCN(c3ccncc3)CC2)=O)=O)CC(N(C)C)C(O)C1 32354,C1(NC(N(C(C)C)C)=O)CCC(C(C)O)CC1.C1(C)C(=O)O1 32355,Cc1cnc(C)c(C(=O)NCC2CCCN2C(=O)CCCNS(C)(=O)=O)c1 32356,c1(-c2nc(-c3scc(C)n3)nn2CC(C)CO)cc(Cl)ncc1Cl 32357,C1(CNC(CC(CCC)CC)=O)CCCC2(CN(C(c3ccnnc3)=O)C2)O1 32358,c1(OC)ccoc1CNC1CC(C(N2CCCC2CO)=O)C1 32359,Cc1c(C(N2CC(NC(=O)C(C)(C)C)CCC2C)=O)cc(Br)cc1N 32360,S(=O)(=O)(C1COC(C)(C)C1)NC(NOCCCNC(=O)OC(C)(C)C)=O 32361,CCN=C(NCc1ccccc1Cl)NC1CCC(C(=O)OC)C1 32362,C12(CNC(=O)Cn3cncn3)CN(C(c3ccc(O)c(F)c3F)=O)CC1CCO2 32363,O=C(N=c1cc(C2CC2)[nH][nH]1)C1CCOCN1C(=O)CC(F)(F)F 32364,N1(C(C(=O)NCC)=O)CC(CNC(C2CCC(N(C)C)CC2)=O)C(O)C1 32365,C12(C(=O)NC(CC=C)CC(F)F)CCCCC1C2(F)F 32366,Cc1cc(C(=O)N(C2CCCC2)CCCNC(=O)C(C)CF)sc1C 32367,C1(N(C)C(c2cncc(C(F)(F)F)c2)=O)CC2CC1N(C(C1CS(=O)(=O)C1)=O)C2 32368,c1(OCCN(C2CCC2)CCOC)ccccc1Cl 32369,N1(C(c2ccc(C(N)=O)nc2)=O)CCN(C(=O)C2=CCSC2)C2CCCCC12 32370,N1(C(C2N(C(c3c(C)oc(CO)c3)=O)CC(=O)NC2)=O)CCOC2(CCC2)C1 32371,C#Cc1ccc(C(=O)NC(C)C(C(C)C)NC(=O)CN(C)CCC)c(F)c1Cl 32372,C1(CNC(C2(COC)CCC2)=O)CCC(C)(C)CN1C(c1ccc(C)nc1)=O 32373,C(C1=NOC2CN(C(C34CC5CC3C4C5)=O)CC12)NC(c1ncc[nH]c1=O)=O 32374,C(=O)(C1Cc2ccccc21)N1C(CN(C)C(c2csc3nnsc23)=O)CCCC1 32375,Nc1[nH]c(=O)c(Cl)nc1C(=O)NCC1CCN1C(c1ocnc1C1CC1)=O 32376,Cc1nc(C(=O)NC2C=CC(CNC(=O)CSC(C)C)C2)c2ccnc-2[nH]1 32377,N1(C(C(C2CN(C(C3CC=C(C)CC3)=O)C2)O)=O)CCC(C)(O)C(O)C1 32378,N#Cc1cnccc1-c1cnc(C(F)(F)F)cc1C(=O)Nc1cc(O)nc(O)n1 32379,CC(CF)CC(=O)NCC1CN(C(c2cnn(-c3cccc(F)c3)c2)=O)C1 32380,n1(CC=C)ccnc1C(=O)NCCCC1CCCN1C(=O)CN(S(C)(=O)=O)C 32381,C(CC(C)C)(C(=O)NC1CN(Cc2ccccc2C(F)(F)F)CC1C#N)NCC 32382,N1(C(=O)Nc2cccc(-c3nccc(C)n3)c2)Cc2c(F)cccc2C(C)(C)C1 32383,C12(NC(=O)CC3COCCOC3)CCCC1CN(C(c1cc(O)nc(O)n1)=O)C2 32384,CC1CCCC(NC(N2CCNC(=O)C2C)=O)CC1 32385,C=CCC(CC)C(=O)N(C1CN(C(C23CCC(CO)(CC2)C3)=O)CCC1C)C 32386,Cc1cc(C(N2CCC(C)(CNC(C3CC4CC3CC4O)=O)CC2)=O)ccc1O 32387,C12(C(N3CCC(O)(C(C)NC(C(=C(C)C4CC4)F)=O)C3)=O)CC3CC1C2C3O 32388,c1(CNC(CN(C(C2CC2C2(C)COC2)=O)CC)=O)nc(C)cc(C)n1 32389,c1(C(C(=O)NC(C(C)C)CNC(c2nnsc2C(F)F)=O)C)cc(F)cc(F)c1 32390,N1(C(C(CSC)C)=O)CCCN(C(c2ccc(C(F)F)c(F)c2)=O)CC1CO 32391,c1(C(=O)NCC#CCNC(=O)CNC(C2CCC2)=O)cn2ccnc2cn1 32392,N1(C(C(C)OC)=O)CCCC(N(C)C(c2ccc(-n3cncn3)cc2)=O)C1 32393,c1ccc2c(c1)CN(C(=O)COC1CCC1)C2.O=C1CC(C(=O)NC2CC2)CCN1 32394,c1(C(=O)NCC(CNC(C(C2CCCOC2)OC)=O)O)c(F)ccc(F)c1F 32395,c1(C(=O)NC2(C)CN(C(c3c(O)cc(C)nn3)=O)C2)cc(F)cc2nccnc12 32396,c1(C(C(=O)NCCC)N(CCN(C)CCO)C(C)C)ccc(SCCCC#N)nc1 32397,C1(C)(CN(C)C)CCN(C(C2CCC(NC(=O)C(C)(C)F)CC2)=O)C1 32398,C1(N(C(c2ccc3occc3c2)=O)CC2N(C)C(=O)CC2)CCCC12CCNCC2 32399,c1(C(=O)NCC(CNC(C2(COC)CCOCC2)=O)C)nc(C)ccc1OC 32400,C1(NC(C2C(O)CCCCC2)=O)C2CC3C1C3C2C(N1CCCC1CN)=O 32401,C(=O)(C(Cc1ccc(O)cc1)C(F)(F)F)NCCCC(C)NC(C(C)=CCC)=O 32402,C(=O)(C1=CCCOC1)NCC1CC(NC(C2CC(OCC)C2)=O)C1 32403,Cc1cc(C(=O)Nc2cccc(CNC(c3scnc3C3CC3)=O)c2)cnc1O 32404,CC1C(C(=O)NC2CCN(C(=O)C=Cc3cnc[nH]3)C2)OC2CCCCC12 32405,CC(=O)CCCC(=O)NC12CCC(C1)N(C(=O)C(C(C)(C)C)OC(C)(C)C)C2 32406,C1(C(N2C(CNC(=O)C(=O)NCC(F)F)C(O)C(O)C2)=O)CCCC(F)(F)CC1 32407,CCC(F)(F)C(C)(C)C(=O)N1CCC(C(C)NC(C2(C#N)CC3CC3C2)=O)C1 32408,c1(C(N2C3CCC(NC(c4cnc(Cl)s4)=O)C(C3)C2)=O)cnc(O)c([N+](=O)[O-])c1 32409,C(=O)(CCNC(c1cnsc1)=O)NC1C(C)C1 32410,c1(NC(C(CCCC)NC(=O)C(F)CC2CCOC2)=O)ccc2c(c1)CCC2 32411,CC(C(C)CO)N(CC(=O)Nc1ccc(Br)s1)Cc1scnc1Br 32412,Cc1cc(C(=O)NOCC(=O)NCc2ccco2)[nH]c1C 32413,N1(C(C(C)CCO)=O)CC(NC(c2ccc3nc(O)[nH]c3n2)=O)C(S(C)(=O)=O)C1 32414,c1(OC)ccc(C(C(=O)NCC(C2CCC2)NC(c2cc(Cl)no2)=O)OC)cc1 32415,c1(C(N(C2CN(C(C3(OC)CS(=O)(=O)C3)=O)C2)C)=O)cc2c(C)c(F)ccc2[nH]1 32416,Cc1cn2ccc(C(=O)NC3CC(CNC(c4sccc4Cl)=O)C(O)C3)cc2n1 32417,N1(C(C2(C)CC2(F)F)=O)CCC2(CCN(C(c3cnc(NC4CC4)s3)=O)C2)C1 32418,N1(C(c2c(C(C)C)nns2)=O)CCCCC1CCN(C)C(C1COCCO1)=O 32419,c1(OC)cc(NC(C2CC2NCc2ccnc(-c3ccccc3)c2)=O)c(C)cn1 32420,N1(C(C)Sc2nnc(-c3nnc(-c4cccs4)o3)s2)C(=O)c2ccccc2C1=O 32421,c1(OC)ccc2c(c1)C(=O)CCN2C(=O)Cc1c(C)nc(C)nc1O 32422,N1(C(C(CC)n2cncn2)=O)C2CCC1CN(C(=O)C=CC1(C)CCOCC1)C2 32423,C1(COC)CN(C(=O)CCc2cnc(O)[nH]2)CCN1C(=O)CS(C)(=O)=O 32424,C(=O)(CN=c1[nH]c(C)cs1)NCC1N(C(c2cc(CSCC)on2)=O)CC(F)C1 32425,c1(C(N2CC(O)(CCNC(C3(F)CCOC3)=O)C2)=O)cc(F)ccc1Br 32426,C1(CNC(c2c(CC)cno2)=O)C(C)CCCN1C(c1cnc[nH]1)=O 32427,N1(C(c2c(C)cc(CNC(C3CC34CCCC4)=O)o2)=O)CCCC2C(=O)NCC12 32428,N1(C(C(C)OCCC(C)C)=O)CCCN(C(=O)C=Cc2cnc[nH]2)CCC1 32429,C1(C(N2CCCC(CNC(C3CCC3)=O)C2)=O)CCC2CC1CO2 32430,C1(CC(=O)N(CCC)CCNC(=O)C2=C(Cl)CC2)CSc2ccccc2O1 32431,C1(NC(CC(C)C(F)F)=O)COC2(C1)CN(C(C1CC=CC1)=O)C2 32432,N1(C(CC2(OC)CC2)=O)CC(NC(=O)CCc2ccc(N(C)C)nc2)C(C)(C)C1 32433,c1(CC)nc(Cl)nc(N2CCC(NC(C3CCC(NC(C)=O)CC3)=O)CC2)c1Cl 32434,N1(C(CC(=O)OCC)=O)CCC(C)C1C(N1CCN(C(C)C)CC1)=O 32435,c1(C(=O)NCC2C(CNC(c3cncc(CO)c3)=O)C2)c[nH]ccc1=O 32436,CC(C)CC(C)(CNC(C1OCCCC1(C)C)=O)NC(=O)CC12CCCC1C2 32437,n1(C)nc(C)c(C(=O)OC)c1C.n1(CCCC)nnnc1C(CC(C)SC)N 32438,O=S(=O)(c1ccc(F)c(Br)c1F)Nc1cccc(-c2ccccc2)c1 32439,C#CCC(CO)NC(C1(CNC(=O)CCOC2CC2)CCC1)=O 32440,C1(CC(=O)NC2CCN(C(C)C)CC2)CC2(C1)CN(C(C1CC(C)(F)C1)=O)C2 32441,C(CC(O)C(=O)NCC1CCCN1C(C1CC(c2cccc(F)c2)(F)C1)=O)SC 32442,C1(NC(c2ccc(C(C)C)cc2O)=O)CN(C(=O)CCS(C)=O)C2(CCC2)C1 32443,c1(OC)cc(C(=O)N(C2CC3(CNC3)C2)CC2CNC(=O)CO2)cc(Cl)c1 32444,c1(CN2CCC(C3N(C(C(CCCC)F)=O)CCC3)CC2)cc(F)c(O)c(F)c1 32445,C12(CNC(C(CC=C)NC(C)=O)=O)CCC(CC1)N2C(=O)C(F)(F)COC 32446,c1(C(C(=O)Nc2ccc(OC)cc2)N(C2CCOCC2C)C)cc(C)ccc1Br 32447,c1(NCC2(O)CN(C)C2)cccc(C(=O)OC(C)(C)C)c1.C12CC(C1)C(=O)N2 32448,CC(C)C(C)CC(=O)N1CC(NC(C2CCC(C)(C)C2)=O)C1 32449,N1(CC(=O)NCCCN(C(C2C(C)COCC2)=O)C)CCCc2sccc2C1=O 32450,c1(C)cccc(C(F)(F)F)c1F.C12CCCN(C1)N(C)C(=O)C2.C1(S)CC1 32451,CC1=C(C)CC(C(N2CCC(C(=O)NC3CNC(=O)C34CC4)C2C(C)C)=O)CC1 32452,NS(=O)(=O)c1ccsc1C(N1CC(O)(CCNC(=O)CC2COCCO2)C1)=O 32453,c1(C(=O)NC(C(=O)NCC2(OC)CC2)C)c[nH]c(=N)c(C)c1 32454,CCC(C)(C)C(O)C(=O)N1CC(C2(NC(=O)C(C)CSC(F)(F)F)CC2)C1 32455,CCC(CC(=O)N1CCC(C)(NC(=O)CCCNC(=O)OC)C1)OC 32456,C1(C(N2C(C(=O)NCCOC(C)=O)CC2)=O)CCC(C2CC2)C1 32457,C(=O)(C(C)(C)CCC)NCCCN1C(=O)C1.C(=O)(CSCC(=O)OCC)NCC=C 32458,N1(C(c2cncc(-c3c(C)ccc(C)c3)n2)=O)CCC2SC(=O)C=C2C1 32459,c1(C(N2C(C)CC(CNC(c3ccnn3C)=O)C2)=O)cccc2c1CCO2 32460,Cc1cc(S(N)(=O)=O)cc(C(=O)NCC(C)N(C(=O)CCCCC#N)C)c1C 32461,N1(C(C2CC3(CC3)CN2Cc2cccc3c2OCO3)=O)Cc2cccc(Br)c2C1 32462,Cc1ccc(-c2cc(C(N3CCCC(N(C(=O)C4=CCCS4)CC)C3)=O)n[nH]2)cc1 32463,C(=O)(N=c1[nH]sc2c(Br)cccc12)NC1(c2ccccc2)CCC(=O)NC1 32464,CCC(F)(F)CC(=O)N1CCCC(NC(=O)CCCn2cccn2)C1C 32465,c1(-c2[nH]c(=N)sc2)ccc(C(=O)NCC2(NC(C3CCOC3C)=O)CCC2)cc1 32466,c1(C(N2CCC(CC(=O)Nc3onc(C)c3Br)C2)=O)cc(F)ccc1[N+](=O)[O-] 32467,CCN=c1ccc(C(=O)NC2CC2NC(c2ccc(C(C)(C)C)s2)=O)c[nH]1 32468,N1(C(C2CCN(C(c3cc(OCC)c(Cl)nc3)=O)CC2)=O)CCCC(F)(F)CC1 32469,C(C(CC(F)(F)F)NC(C1(F)CCCC1)=O)NC(CSCCCC)=O 32470,C1(NC(=O)NC2(CC)CCNC2=O)CC2(CC(OC)C2)C1 32471,C(=O)(C(C)S(N)(=O)=O)N1CCN(CC(=O)Nc2ccc(CCCCC)cc2)CC1 32472,C=CCC(CC(F)F)C(=O)N1CCN(C(=O)CCC(CC)CC)C(CC(F)F)C1 32473,N1(C(C2C(C)(C)CC2)=O)CCC2(CCN(C(c3cnc(C(N)=O)cn3)=O)CC2)C1 32474,c1(C(=O)NCC(CNC(c2csnn2)=O)CO)ccc(-n2cncn2)cn1 32475,N1(C(c2ncn(C)n2)C(=O)NC2CCOC2)CCC(CC2(O)CC2)CC1 32476,N1(C(C=CC(C)=O)=O)CCC(CC(C)(C)NC(=O)Cc2nccn2C)CC1 32477,CC1CN(C(=O)COCCO)CC1NC(=O)C(C)Cc1cccc(N(C)C)c1 32478,c1(C(=O)OCC)cc(C(=O)NC(C)CC(C)NC(C2(F)CCCC2)=O)[nH]n1 32479,c1(C(=O)NCC(CC)NC(C2CCN(C)C2)=O)nncc2ccccc12 32480,Cc1nn(CC(N2CC3(CC(NC(C4(CF)CC4)=O)CO3)C2)=O)c(C)c1[N+](=O)[O-] 32481,c1(OC)ncnc(C(=O)NCCCOCCNC(C2CCNC2=O)=O)c1F 32482,Cc1ccc2ncc(C(N3CCC(C)C3CNC(=O)C(C)(C)CC(F)F)=O)n2c1 32483,C1(NC(c2c(C)nn(C)c2F)=O)COC2(CCN(C(=O)CS(=O)(=O)N(C)C)C2)C1 32484,CCCC(CCNC(C1CCC1CNC(C1(OC)CCOC1)=O)=O)CCC 32485,CCCC(CCC)CC(=O)NC(c1cn(C)nn1)C(N1CCC(O)CC1)=O 32486,C(CCCCCC(=O)NC1(CC2CC2)CC1)NC(c1n(CC)ccc1)=O 32487,c1(N2CCC=C(C(=O)NCc3cc(C)c(O)c(C)c3)C2)ccnc(S(C)(=O)=O)n1 32488,C1(CCC)(NC(c2cccc(N(C)C)n2)=O)CCCN(C(=O)C(C)C(F)F)C1 32489,c1(C(=O)NC2CC(CNC(COC(CC)(C)C)=O)C2)cc(OC(C)C)ncc1Cl 32490,N1(C(Cc2c(C)nc[nH]2)=O)CC(NC(=O)C2=CCOCC2)CC12CCOCC2 32491,n1(CC(N2CCC(CNC(CCC(=C)C)=O)(OC)C2)=O)ccc2c(C)cccc12 32492,c1(C(=O)NC(CNC(C(C)c2ccsc2)=O)C2CC2)ccc(Cl)c(F)c1O 32493,C1(C)(NC(CN(C2CCC2)C(C2C(C(C)C)CCC2)=O)=O)CN2CCC1CC2 32494,Cc1cnccc1C(C)C(=O)NCCN1CCC(NC(=O)C(N)=O)CC1 32495,c1(COC)cccc(C(=O)NC(C)C(C)NC(C2(C(F)(F)F)CC2)=O)c1 32496,n1(C(C)C)cnc2c(N(CCCN)C)nc(N3C4CCC3C(C)C(=O)C4)nc12.C=O 32497,c1(C(=O)NCCOCCCNC(C2(C(=O)NC3CC3)CC2)=O)csc(Cl)c1 32498,C1(C(=O)NC(CC)CNC(=O)CCN(S(C)(=O)=O)C)CCOC1CC 32499,C1(O)(C(N2CC(C)SC2)=O)CCCC(C)CC1 32500,C(=O)(C(C)(C)C(=O)NC1CN(C(=O)CC(=O)OC(C)(C)C)CC1C)NC 32501,c1(CN(CCOC)CCNC(c2coc(CC3CC3)n2)=O)nn(C)c2c1CCC2 32502,Cc1c(C(=O)NC2CCCC(NC(c3occc3F)=O)C2)ccn1C(C)C 32503,Cc1cccc2c1CC(C(=O)NCC(CC(C)C)NC(=O)C(O)C1CCC1)N2 32504,c1(CNC(c2cc(C(=O)OC)n(C)c2)=O)ccc([N+](=O)[O-])cn1 32505,c1(NC(N2CC(SC)CC23CCC3)=O)cnc2ncccc2c1 32506,c1(C(=O)NC2(CN(C)C(c3cc(F)c[nH]3)=O)CC2)cc(O)nc2[nH]c(=N)ccc12 32507,N1(C(c2cc(C)n(C(F)F)n2)=O)CC(N(C(=O)CCOC2COC2)C)C(C)(C)C1 32508,N1(C(C)=O)CC2CC1CN(C(=O)C(C(C)C)NS(=O)(=O)c1cnn(C)c1)C2 32509,C1(CCC)CN(C(c2cc(Br)c(Br)o2)C(=O)NCc2nnn(C)n2)CCO1 32510,N1(C(C2CC(=C)C2)=O)CC(CNC(=O)C=Cc2cc(Cl)sc2Cl)OC(C)(C)C1 32511,C1(NC(CCC(=C)Cl)=O)CC12CCC(NC(c1ccsc1)=O)CC2 32512,CC1CC(=O)NCC1C(=O)NCC1CN(C(C2SCCCS2)=O)CCCO1 32513,N1(C(=O)OC(C)(C)C)CCCC(CCCCNc2cccc(C(N)=O)n2)C1 32514,C(=O)(CCC(=O)NC(CNC(c1sc(N(C)C)nc1Cl)=O)C1CCC1)OC 32515,C1(CNC(C2CCCC(C(N)=O)C2)=O)(NC(c2cc(F)n[nH]2)=O)CCCCCC1 32516,C1(NC(C#CC(C)C)=O)CCCC2CN(C(c3coc(C(C)(C)C)n3)=O)CC12 32517,C1(C(N2CC(C)(CNC(=O)CC3CCC3)OCC2)=O)OCC2CCCC1C2 32518,CC1CC(NS(=O)(=O)c2ccccc2COCN2C(=O)CCC2=O)c2nccn21 32519,N1(C(C2(CC#C)CCCCO2)=O)CCCCCC(NC(c2ccoc2Cl)=O)C1 32520,C(CC(C)(O)COC)N.C(=O)(CC(C)(C)O)C(=O)CCN 32521,c1(C(=O)NC23CC2CN(C(=O)CCCn2cncn2)C3)ccn2ccsc12 32522,N1(C(Cn2ccc(C)n2)=O)CCC(NC(=O)Cc2ccccc2Cl)C(C)C1 32523,N1(C(C(CC)C)=O)CCN(C(=O)CCCCCF)C(CC(=O)NC)C1 32524,Cc1cnc(C(=O)NC(C)C(C)NC(=O)Cc2cnc(C)[nH]2)c(Br)c1 32525,N1(C(C(C)(C)C2CCOCC2)=O)CCC2(COC(CNC(=O)CC3CSC3)C2)C1 32526,c1(C(N2CCC(C(=O)Nc3cc(C)c(O)cn3)C(O)C2)=O)ccccc1[N+](=O)[O-] 32527,C1(NC(Cc2ccn(CC)n2)=O)CCN(C(C2COCCN2C)=O)C1C1CC1 32528,C1(CCC(=O)NCC(CC)NC(C2CSCN2C(C2CCC2)=O)=O)CCC(=O)N1 32529,CC(C)=C=CC(=O)NCCC1(C(=O)N(C(C)CC(F)(F)F)C)CC1 32530,C(c1ccnc2ccccc12)=CC(=O)NC1CCCC1NC(C1CC2CC2C1)=O 32531,S(=O)(=O)(c1cncc(Br)c1)NC1CN(C(=O)Cc2ccccn2)CC1F 32532,N1(C(c2cc(C)[nH]c2)=O)CC=CCC1C(=O)NCC1CC=CCC1 32533,c1(C(N2CC(CCNC(CS(CC)=O)=O)C(C)C2)=O)ccc(C)cc1C 32534,c1(CCC(=O)N(C)CCOCCN(C(=O)CCC2CCOC2)C)cccnc1 32535,CC1CCC(C(=O)NC2(CCNC(=O)CCNC(=O)C(C)(C)C)CCC2)S1 32536,c1(OC)ccc(S(=O)(=O)N2CC3CN(Cc4ccc(C)c(F)c4)CC3C2)cc1 32537,C1(C(N(C(CCNC(C(C)(C)SC)=O)C)C)=O)CCCN(C(=O)OC(C)(C)C)C1 32538,N1(C(c2c(CC)nns2)=O)CCC(C)(C)C1C(=O)NCCc1ccc(C)cc1 32539,c1(C(=O)NCCCNC(C(C)OCCC=C)=O)ccc(F)c2[nH]ccc12 32540,c1(C(=O)NCC2(O)CN(C(c3ncnc(C)c3C)=O)C2)cc(F)cc(Cl)c1N 32541,CC1CN(C(C2CNC(=O)O2)=O)CC(C)N(C(=O)C2=NNC(=O)CC2)C1 32542,C1(CN(C(CCC2CCCC2)C(=O)NC2CC(F)(F)C2)C)CCCN(C)C1=O 32543,c1(OC)ccc(CCNC(=O)C(N2CCN(CC(C)O)CC2)=O)cc1OC 32544,Cc1ccc(C(F)F)c(C(=O)NCCCCN(C)C(C2(C)CCCS2)=O)c1 32545,N1(C(c2c(C#C)c[nH]n2)=O)CC(F)(F)CC1(C)CNC(c1c[nH]cc1C1CC1)=O 32546,C=C=CC(C)C(=O)NCC(C)N(C(C1COC(=O)N1)=O)CC 32547,Nc1cc(C(=O)NCC2(NC(c3nc(C4CC4)cs3)=O)CCC2)cc(F)c1 32548,c1(OC)cc(C(=O)NCC2CCN(C(C3CCC=CCC3)=O)C2)cc(C2CC2)c1 32549,Cc1c(C(=O)NCC23CC(NC(=O)Cn4cc(Cl)cn4)(C2)C3)cccc1Cl 32550,c1(COC)nn[nH]c1C(=O)NCCCN(C(c1ccc(C(N)=O)s1)=O)C1CC1 32551,N1(C(C)=O)CCc2cc(C(N(C)C(N3CCC4CCC34CN)=O)=O)ccc21 32552,N(C1Cc2ccc(F)cc21)C(=O)C=Cc1ccc(Cl)c(Cl)c1 32553,C1(n2c(C(c3nc[nH]n3)NCc3cnc(CCOC)[nH]3)nnn2)CCCCCC1 32554,C12(CNC(c3n(CC)ncc3)=O)CC(CO1)N(C(=O)C(C)OCC(C)C)C2 32555,C1(C)(CNC(c2c(OC)nsc2OC)=O)CN(C(=O)CCC(N)=O)C(C)(C)C1 32556,C(CN=c1cc[nH]cc1S(=O)(=O)NCC1(CO)COC1)OC 32557,C(=O)(C(=O)C(C)(C)CC)NC(COCC)C(=O)NCC1(CO)CCCO1 32558,Cc1cc(C(=O)NCCC2CCC(NC(c3nc(C)n(C)c3C)=O)C2)nc(O)n1 32559,C(=O)(C(C(C)(C)C)C1CCCC1)N1C(C2(NC(CCOC(C)C)=O)CC2)CCC1 32560,C1(C2CCCO2)(C(N2C(CNC(C=C(C)C3CC3)=O)CC2)=O)CCCO1 32561,N1(C(=O)OC(C)(C)C)CC2(CCOCC2)C1C(F)(F)F.C12CCCC1NC(=O)N2C 32562,C1(C(=O)OC)CC(F)(F)CN1C(C(=O)NCc1cccs1)C1CC1(C)Br 32563,C(=O)(CC1=NNC(=O)C1)NC(C)(CNC(C1CC(CC2CC2)C1)=O)C1CC1 32564,C1(C2(C)CC2)(C(=O)NC(C2C(C(N(CC#C)CC#C)=O)C2)C)CC1 32565,c1(N(C)Cc2c(C)cccc2F)cccc(S(=O)(=O)N2CCC(C(C)C)C2)n1 32566,CCC(CC(=O)NCCc1ccc(CNC(=O)C=CBr)cc1)C(F)F 32567,c1(C(=O)NC(C(CO)NC(c2c(C=C)cnn2C)=O)C)c(F)cc(F)cc1Cl 32568,c1(C(=O)NC2CC(c3ccc(Cl)cc3)(O)C2)cnn2c1OCC1(COC1)C2 32569,N1(C(Cc2ccn(C)n2)=O)CCOCC1CNS(=O)(=O)CC1CC1 32570,C1(CCC)C(=O)NCCN1C(=O)C(C)(CSC)NC(C1C2CC(=O)CC12)=O 32571,c1(OC)ccc(CO)cc1NC(C1CCN1C(c1ccccc1OCF)=O)=O 32572,N1(C(C(c2cc(C)c(F)cc2)=O)=O)CC2CN(C(=O)C(O)O)CC2C1 32573,Cc1ccc2c(c1)C(C(=O)NC1CCC(NC(=O)COCC3CCCC3)C1)C2 32574,CS(=O)(=O)CCC(C(N)=O)NC(=O)CCc1cccc(F)c1Br 32575,C1(CNC(C(C)CNC(=O)Cc2ccc[nH]2)=O)CC12CCOCC2 32576,c1(C(=O)NCC(=O)N(C2CC(C)(C)C2)C)c(F)cccc1F 32577,c1(C(=O)NCC2(CN(C(C(CC=C)CC)=O)C)CC2)ccc(Cl)c(OC)c1F 32578,CCC(C(=O)NCCN(C(=O)C(C)C1CCCC1)CCCN(C)C)C(C)C 32579,Cc1ccc(C(N2CCC2C(=O)NCCCS(C)(=O)=O)=O)c(O)n1 32580,N1(C(C2CC(SC)C2)=O)CCCC(C2CC2NC(c2cccc3cc[nH]c23)=O)C1 32581,c1(NC(C2CC2C(=O)NCCCc2cccnc2)=O)cc(Br)cc2[nH]ncc12 32582,c1(C(=O)NC2CCC(C)(OCC)CC2)ccc(F)c2c1CCC2.C12CC1C(=O)N2 32583,CC1(C(N2CCN(C(=O)CNC(c3ccc(=N)[nH]n3)=O)CC2)=O)CCCS1(=O)=O 32584,C1(C(=O)NC2C(NC(c3ccc(OC)c(O)c3)=O)CCC2)Cc2cccnc2C1 32585,Cc1cc(C(=O)N(CCNC(=O)C(CO)N(C)C)C2CC2)nc(C)c1 32586,C1(NC(Cc2nc(C)[nH]n2)=O)CC2CCC1(N=c1[nH]nc(C3CC3)s1)C2 32587,C1(NC(C2(C)CCNC2=O)=O)CCCN(C(C2CC(F)(F)CS2)=O)CC1 32588,c1(CN(CCCn2cc(SCC(=O)OC)nn2)C2CC2)cccc(Br)c1[N+](=O)[O-] 32589,N1(C(C2N(C(CC(CC)SC)=O)CCC=C2)=O)CCC(C)=C(F)C1 32590,C1(CNC(CS(CC)=O)=O)CC(C)(C)CN1C(c1ccc(SC(F)F)cc1)=O 32591,Cn1ncc2nc(Cl)nc(NCC34CCC3CN(C(=O)CC3(C5CC5)CC3)C4)c12 32592,C1(C(=O)NC(C(=O)OC)C)CC12CC(NC(=O)Cc1cn[nH]c1)C2 32593,C1(C)(C(N2CCC(C(C(=O)NCCc3c(C)nc[nH]3)C)C2)=O)CCN(C)C1 32594,c1(N2CCN(C(C(=O)N(CC#C)CC=C)C)CC2)ncnc2sc(C)nc12 32595,c1(C(C(=O)NC(C(C)C)CNC(C2CC3CC3C2)=O)(C)F)ccccc1F 32596,c1(OC)cccc2c1CNC(C(N1CCC(n3cc(Cl)cn3)C1)=O)C2 32597,C(=O)(CC(Cl)Cl)NC1(C(=O)NCCC2(COC)CC2)CSC1 32598,O=S(=O)(C=Cc1ccccc1)NCC12CC1CN(S(=O)(=O)c1ccc(O)cc1)C2 32599,c1(C(=O)NC2(CNC(C(CC#C)O)=O)CCCCC2)ccc(F)c(O)c1F 32600,CCCCCCC(CC)C(=O)N1CC(C)(NC(c2cccc3c2ccn3C)=O)C1 32601,c1(OC)ncc(C(=O)NCC(C2CC2)NC(C2CCC(C(N)=O)N2C)=O)cc1Cl 32602,N1(C(C2(C(=O)N(C)C)CC2)=O)C(C(=O)OC(C)(C)C)CCC1(C)C.C12CC(C1)N2 32603,Cc1nc2ccc(C(N3CC(NC(C4CCC(=O)O4)=O)C3)=O)cc2n1C 32604,c1(-n2c(C(CC)CC(C)C)nc(C3CCCS(=O)(=O)C3)n2)nc2cc(Cl)ccc2s1 32605,n1(C(C)C)ccc(C(=O)NCC(C)N(C(=O)C(C)NC=O)C)n1 32606,N1(C(c2sc3cc(C)sc3c2)=O)CCC(C2CCN(C(=O)CC#N)CC2)C1 32607,C1(O)(CNC(C2(C(C)C)CC2)=O)CCCN(C(c2ccc(O)cc2Cl)=O)CC1 32608,C1(CNC(c2cncn2C)C)CNCCC1c1ccc(F)cc1 32609,N1(Cc2c(OCC=C)cccc2)CC2CN(C(C3CC4CCC3O4)=O)CC12 32610,C1(CNC(C(C)SCCCC)=O)C2CN(C(=O)C(C)Sc3ccc(F)cc3)CC12 32611,n1(CC)cc(CN2CC(O)CC2C(=O)Nc2cc(O)ccc2Br)c2cccnc12 32612,CCC(F)(F)CC(=O)N1CCOC(C(N2CCCC3CC23)=O)C1 32613,N1(C(C2C(C)(C(F)F)C2)=O)CCN(C(=O)CCC2CC2)CC12CC2 32614,c1(-c2onc(COC)n2)cccc(CNC(=O)CC2(C(=O)O)CCCC2)c1 32615,N#Cc1cccc(Cl)c1NC(C1CN(Cc2nc(Cl)ccc2Cl)CCO1)=O 32616,Cc1cnn(C)c1C(N1CC(C)(NC(=O)C(C)c2cncs2)C1)=O 32617,Cc1cnc(C=CC(=O)NCCC2CCCCN2C(C2C3COCC23)=O)[nH]1 32618,C=C(Cl)CCC(=O)N1CC(CCNC(C2CC3CCC2C3)=O)(OC)C1 32619,C1(C)(C(=O)NCC2N(C(CCC(C)C#N)=O)CC2)CCCCNC1=O 32620,c1(CNC(N)=O)ccc(C(N2CC(O)(CNC(=O)CC3CCSCC3)C2)=O)cc1 32621,c1(C(N2CCN(C(c3cn4c(n3)CCC4)=O)C3CC23)=O)ccc(F)c(Br)c1 32622,C(=O)(C1=CC(C)(C)C1)NC(C(c1c(OC)cccc1)NC(C1(SC)CC1)=O)C 32623,C1(CNC(c2c(C)scc2)=O)CCN(C(=O)C2=CCOC2)CC1C 32624,c1(C(=O)NCCC2CCN(C(C(N=S(C)(C)=O)=O)=O)C2)cnc2ncnn2c1O 32625,C=CC(CC)CC(=O)N1CCN(C(=O)CN2CCCCC(=O)C2=O)C(CCO)C1 32626,c1(CC)nn(C)c(CC)c1C(=O)NCC=C1CCN(C(=O)C(C)S(C)(=O)=O)CC1 32627,c1(NCC(N2CCCC(CS)C2)=O)ccc[n+]([O-])c1 32628,N1(C(C=CC(CC)C)=O)CCN(C(c2cnncc2O)=O)C(C)C1C 32629,C1(C2=CCCCCC2)(C(N(CCCNC(c2c(C)onc2CO)=O)C)=O)CC1 32630,C1(N(C(CCN(C(=O)CC=C(C)C)CC=C)=O)C)CCCC(O)C1 32631,c1(C(N2CCCC(NC(C3=CC(C)(CC)C3)=O)C2)=O)cc(C#N)c(O)nc1N 32632,N1(C(C2N(C(C)=O)CCC2)=O)CCC12CN(C(=O)CCCn1ccnn1)C2 32633,N1(C(C2=CCC(NC(C(C(C)C)=O)=O)C2)=O)CCn2ccnc2C1 32634,N1(C(C(C(=O)OCC)OC)=O)CCC(O)(CC(=O)NC2CCN(C(C)=O)C2)CC1 32635,c1(CC(=O)N(CC(=O)NC(C)Cc2ncn(C)n2)CC#C)cccc(C)n1 32636,Cc1c[nH]c(C(=O)N(C(CCC(=O)NCC(C)C(C)C)C2CC2)C)c1C 32637,c1(OC)cc(O)ccc1NC(c1cnc(C2CC2)nc1C)=O 32638,c1(CC(N2CC(N(C(C(C=C)O)=O)C)C(C)(C)C2)=O)cnc2ccccc2c1 32639,C1(C(=O)NC2C=CCN(C(c3ccccc3Br)=O)C2)CC2CC(O)C(C1)C2 32640,C=CCCCC(C)(C)CNC(c1cn(CCNC(=O)C(F)CC2CCOC2)nn1)=O 32641,N1(C(C(CC)(C)COC)=O)CC2C1CCCN2C(c1cc2ccsc2n1C)=O 32642,Brc1ccc2c(c1)ncn2CCNC1(CCc2nn[nH]n2)CCNCCC1 32643,C1(CN=C(NC(C=C)C)NCc2nn(CC)cc2Br)CC(S(C)(=O)=O)C1 32644,C12(CC(=O)NCC3(COC)CCCC3)CCC1CN(C(=O)C1=CCCCC1)C2 32645,c1(C(N2CC3CC3(NC(C3(CF)CC3)=O)C2)=O)ccc(Cl)cc1Br 32646,c1(C(=O)NC(CC)CN(C(=O)Cc2ccoc2C)C)occ(C)c1C(=O)OC 32647,C(=O)(CC(C)C1CC1)NCCC(C)NC(=O)C(c1ccncc1)C 32648,N1(C(CC2CCN(C)CC2)=O)CC2(NC(C3COC(=O)N3C)=O)CCCC2(F)C1 32649,c1(OC)cc(OC)c(C(N2CC(NC(=O)C(C)CF)C(O)C2)=O)c(N)c1 32650,Cc1cc(Br)c2ncnc(N3CCCC(c4n[nH]c(C)n4)C3)c2c1 32651,Cn1cc(Cl)cc1C(c1nnnn1CCN1CCOCC1)NCC1CC(C)(C)CO1 32652,c1(C(=O)OC)cc(C(=O)NCc2cccc(-c3ncc(C)o3)c2)c(C)s1 32653,N1(C(c2ccc(CSC)o2)=O)CC2CCC(C1)N2C(=O)CCC1CCCO1 32654,n12nnc(n1)CNC(=O)C2.N1(CC)CCCC1C(=O)OC(C)(C)C 32655,C1(CNC(CCN(C(COC(C)C)=O)CCCO)=O)CC=CCC1 32656,CC1CC(NC(c2ccc(Br)c(O)n2)=O)CN(C(C2CCC(=O)C2)=O)C1 32657,N1(C(C(C=C)(C)C)=O)CCC(NC(c2ccc(OC)cc2OC)=O)C(C(C)C)C1 32658,C(=O)(C(F)(F)CCn1ccnn1)NC(CC(C)NC(=O)CC1CC(O)C1(C)C)C 32659,C1(NC(C(C)=C2CCCC2)=O)CCN(C(=O)C=Cc2ccncc2)C1C 32660,C1(NC(COC)=O)C2CCCN(C(=O)CN3CC(C)(C)C3)C2C1(C)C 32661,Cc1cccc(-c2cc(C(=O)N(C(C)CNC(C3(C(C)(F)F)CC3)=O)C)on2)c1 32662,C12(C(=O)NCC3CC4(CCC4)CO3)CC(CN(C(c3nn[nH]n3)=O)C1)C2 32663,n1(CC)nc(C)c(C(N2CC(NC(C3(O)CCSC3)=O)C(SC)C2)=O)c1Cl 32664,C1(N2CCOCC2)(C(N(CCN(C(C)=O)CC)CC)=O)CCCC1 32665,C(C)(CO)(C(=O)NCCC(O)CO)N(C)C(C1CC1c1ccoc1)=O 32666,C1(CNC(=O)C=Cc2ccoc2)CC2CCC1N2C(=O)CCc1cccc(F)c1 32667,c1(CCC(N2CC(C)(NC(C3C4CC4C4CC34)=O)C2)=O)cnc2ncccn12 32668,N1(C(c2n(CCC)ncc2)=O)CCN(C(=O)CS(=O)(=O)N(C)C)CC(CO)C1 32669,Cc1ncnc(O)c1CC(N1CCC1CNC(C1(O)CC(F)(F)C1)=O)=O 32670,C1(C(=O)NCCC(C)NC(C2(CCF)CC2)=O)OCC2COCCC12 32671,C1(CCC(N)=O)C(=O)N2CC(C)(C2)c2cn1nn2.C1(C(C)C)CC1C(F)(F)F 32672,Cc1c(C(N2CC(O)(CNC(C3CCN(CC(C)C)C3)=O)C2)=O)c(Cl)nn1C 32673,N1(C(C2(C)CC2)=O)CCC2(COCCN2C(=O)C=CC2CCCCC2)C1 32674,C1(CNC(C(C)OCC(C)C)=O)CC(C(=O)NCC2CCCC2N(C)C)CO1 32675,n1(C(C)C)ccc(CC(N2CC(NC(c3ccsc3Br)=O)C2)=O)n1 32676,Cn1cc(C(=O)NCCC2(CNC(=O)Cn3ccc(Br)n3)CC2)nn1 32677,CCC(C)N(OC)C(=O)C1COC(CNC(=O)C(C)CC(N)=O)C1 32678,N1(C(C(CCF)NC(=O)CC2CCC(O)C2)=O)CCOC2(CCC2)C1 32679,N1(C(Cn2ncc(CC)c2)=O)CC(C2CC2C(=O)NC2CCN(CCCO)C2)C1 32680,c1(C(=O)NCCNCC(C2CCCO2)O)cncc([N+](=O)[O-])c1 32681,c1(C(N(CCNC(c2c(CC)onc2)=O)C(C)C)=O)cc2cccn2cn1 32682,N1(C(C(C)NC(C)=O)=O)CC(CNC(=O)Cc2cncn2C2CC2)C(C)C1 32683,c1(CC(=O)NCC2CN(C(c3c(Cl)ccc(N)c3)=O)C2)noc2ccc(F)cc12 32684,C(CC(C)C)(C(=O)NCC(c1ccccc1)CNC(=O)CSc1ccncc1)OC 32685,C(=O)(CCC(C(C)C)NC(c1cc(C(C)C)[nH]n1)=O)NC(C(=O)NCC(C)C)C 32686,C(=O)(C#CC1CCCOC1)NC1CC2CN(C(Cc3n(C(C)C)cnn3)=O)CC21 32687,c1(NCCOC)nnc(N2CCN(CC3CCCC3)CC2)n1C(C1CCOC1)C 32688,c1(CC(=O)NCC2(C(C)(C)O)CN(C(C(F)OC)=O)C2)ccc(F)c(F)c1 32689,C1(CNC(C)CN(C(=O)CCCn2c(O)nnc2O)C)CSc2ccccc2O1 32690,C(C(C(=O)N1CC2CC2C1)C(C)C)NC(CSCCCC)=O 32691,c1(N2C(CNC(=O)Cc3cnsc3)CC2)cc(C2CC2)ncn1 32692,C1(C(=O)NCCC(C)NC(C2CC(=O)N(C)C2)=O)CC(C)(C)C1C(F)(F)F 32693,N1(c2n(C)nnn2)CCOC2(CCCN(C(=O)C(F)C(F)(F)F)C2)C1 32694,CC(O)C(C)(C)C(=O)N1CCC(OCC(=O)Nc2cnn(C)c2C2CC2)C1 32695,C1(C(C(C)(C)C(N)=O)c2ccccc2)CC2(CCC2=O)C1.C12C3CN(CC13)NC2=O 32696,N1(C(CC2CCC(OC)CC2)=O)CC(C2CN(C(=O)C(C)(CO)OC)C2)C1 32697,N1(C(c2cnc(-n3cccn3)s2)=O)CC2(CC(C(F)(F)F)C2)C1 32698,N1(C(C(C(C)C)N(C)C)=O)CC2(CC(CNC(=O)Cc3cnn(C(F)F)c3)C2)C1 32699,c1(C(=O)NCC(CNC(C(C)CN2CCCCC2)=O)CO)cccc(N)c1F 32700,N1(C(CC(C)SC)=O)CCN(C(c2cc(C)on2)=O)CC1c1cc(F)ccc1F 32701,C=CCC(C(=O)NCCCN1CCC1)NC(C1OCCOC1C)=O 32702,c1(C(=O)OC)c(NC(C2CCCN(Cc3nccs3)C2)=O)sc(C)c1C 32703,CC(C)CC(C)CC(=O)N1CC(C)(C)CC1CNC(=O)CC1CCC(C2CC2)O1 32704,Cc1ncc(Cl)c(C(=O)NCCC2(C)CCN(C(=O)CN3CCN(C)CC3)C2)n1 32705,Cc1cc(C(=O)NC2CCC2CNC(C2(N=[N+]=[N-])CC2)=O)cnc1C(F)F 32706,c1(C(=O)NCC2C3(CN(C(c4nc(C)oc4)=O)C3)CC2)cc2n(n1)CCCC2O 32707,c1(C(=O)NC(C2(O)CCN(C(C3CC(C#N)C3)=O)CC2)C)ccc2c[nH]nc2c1 32708,c1(C(=O)NC2(C(=O)NCCC(O)C3CC3)CCCC2)cccc2[nH]ccc12 32709,c1(OC)nccc(C(N2CC(NC(=O)C(C)C)C(C)C2)=O)n1 32710,CC1CCC(C)(C)N1C(C1CCN(c2ccncn2)CC1)=O 32711,c1(CCC(=O)OC)ccc(NC(=O)C(=O)NC(C2CCC(C)C2)C2CC2)cc1 32712,CC1CCN(C(C2CC(O)(C#N)C2)=O)C(C)C1NC(C1CN(C(N)=O)C1)=O 32713,c1(C(=O)NCC23CN(C(CC(=O)OCC)=O)C(CC2)C3)nc2cc(F)ccc2s1 32714,C1(C(C(C)NC(=O)N(C)Cc2ccco2)(C)C)Cc2ccccc2O1 32715,CC(C)(O)C(F)C(=O)NCC1CN(C(C2CC(=O)N2)=O)C1 32716,c1(C(N2CCN(c3nc(C)cc(SC)n3)CC2C)=O)ccnc2c1OCO2 32717,c1(CC)ccccc1-c1cn(CC2CCCC2NC(c2cnn(C)c2)=O)nn1 32718,c1(C(=O)NC(CNC(c2ccc(C)nn2)=O)C2CCC2)c(C)nn(C(C)C)c1C 32719,c1(CN(C(CCC)=O)C)cnn2c1CN(C(=O)C(C)SC)CC2 32720,CC1CCC(NC(c2cccnc2O)=O)CN1C(=O)CC1(NC(C)=O)CC1 32721,CC(CN=c1[nH]c(=NCC2CCC3(CCC3)O2)[nH]c2c1CCCC2)C1CCCC1 32722,C1(NC(C2CNC(=O)N2)=O)(CNC(C2CSCCS2)=O)CCC(F)(F)CC1 32723,C1(CNC(C(=O)NCc2n(CC(C)C)ncc2)=O)CCC2(CO1)CC(O)C2 32724,C12CCC(c3ccccc3)N1S(=O)(=O)C2.C(C1=CCNCC1)N(CC)CC 32725,N1(C(c2nc(C(C)C)sc2)=O)CCCC1(C)CNC(=O)COC1CCCOC1 32726,CC1(C)CC(C(N2CCN(C(=O)C=Cc3ncc[nH]3)C(CO)C2)=O)C(C)(C)O1 32727,C12CCCC(C1)NC2=O.C1(CC#N)CN(C(=O)CO)C1 32728,C1(C2CN(C(CCOCCOC)=O)C2)CCN(C(c2cccnn2)=O)CC1 32729,c1(C(=O)NCC2C(NC(c3c(N)n(CCO)nc3)=O)CC2)cccc2sccc12 32730,c1(C(N(CCN(C(C2(O)CC3CCC2C3)=O)CC)CC)=O)ccc2cn(C)nc2c1 32731,CCCCC(O)CC(=O)NC(C(N1CCCC(C)C1)=O)C1CC1 32732,N1(C(C2CCC(=O)N2)=O)CCCN(C(C23CCC2C3)=O)CC1 32733,C1(NC(CC(COC)C)=O)CC2CC1CN(C(c1ccncc1Br)=O)C2 32734,C(c1ccc(C(F)F)o1)=CC(=O)NCC(CCNC(Cc1cn(C)nc1)=O)O 32735,N1(C(CC)=O)CCc2nc(C(N3CCC(N(C)C(=O)C4CC4)CC3)=O)cn2CC1 32736,C=C(C)C1OCCC1CNC(=O)C(C1CCCCC1)NC(C1CN(C2CC2)C1)=O 32737,N1(C(C(N2CCCC(C)C2)=O)=O)CCCC(C)(CNC(c2ncccc2Cl)=O)C1 32738,CC(CCCc1ccccc1)C(=O)N1CCC(N(C(=O)C2=C(Cl)CC2)C)CC1 32739,c1(OC)cc(C(N2C3CCC2C(NC(=O)CC2CCCCC2)C3)=O)c(Cl)cc1Cl 32740,Cc1ccc(F)cc1C(N1CCC1CNC(C1(F)CCCN(C)C1)=O)=O 32741,C(=O)(C1=NOC(CNC(=O)CC(C)n2ccnc2)C1)NC1(C(COC)O)CC1 32742,Cc1cc(CC(=O)NC2COCC2NC(=O)CC(C)F)ccc1CO 32743,C1(C2=CCOCC2)(CNC(c2cc3c([nH]2)CCCC3)=O)CC1 32744,C(=O)(C(CC(F)(F)F)c1ccc(F)cc1)NCCc1scc(C)n1 32745,c1(C(=O)N(C2(O)COC2)C(C2CC2)C2CC2)c[nH]nc1-c1ccccc1 32746,Cc1ccc(CC(=O)NC2CC(NC(=O)C(C)(C)OC(C)C)C23CCC3)cc1O 32747,c1(CC)nc(C)c(C(=O)NC2CCCC(NC(=O)CCC#N)C2)c(C)n1 32748,C1(CNC(=O)NC(C#CC)(C)C2CCC2)(CNC(=O)OC(C)(C)C)CCC(=O)N1 32749,c1(CC)nc(C)c(CC(=O)NCCCCNC(C2CS(=O)(=O)CCO2)=O)c(C)n1 32750,c1(OC)ccc(CC(=O)NCCC2CCCC2(C)C)c(O)c1 32751,N1(C(C2N(CCCC)CCCC2)=O)CC(NC(c2cc(C)[nH]c2C)=O)C(C)(C)C1 32752,C(=O)(C1=CCCN(C(=O)CC=C(Cl)Cl)C1)N1CC(C)(OC)C1 32753,C1(C)(C(N(C(N(CC(C)O)C(C)C)=O)C(C)C)=O)CCN(S(C)(=O)=O)CC1 32754,c1(C(=O)NC(CC)CNC(=O)C=CS(C)=O)cnc2cnc(Cl)cc2c1 32755,N1(C(c2c(C)coc2)=O)CCC2(CCN(C(=O)CC3COCCOC3)C2)C1 32756,c1(C(=O)NCCC(C)Nc2nccn3nnnc23)cncc2nc[nH]c12 32757,C=C(Cl)C(C)(C)C(=O)NCC(C1CCCN(C(c2ncncc2F)=O)C1)(C)O 32758,C(CC(O)CNC(c1n[nH]cc1Br)=O)NC(=O)COCC1CCCC1 32759,c12conc1CCNC2c1nnnn1C1CC1.C=CCSCC=C 32760,C1(NC(c2cc(F)c(Cl)cc2F)=O)CCCCCN(C(c2cc(CO)[nH]n2)=O)C1 32761,C=CCC(CC(F)F)C(=O)NC(CNC(c1cc(CC)cc(N)c1)=O)C(C)(C)C 32762,c1(C(N2CC(CNC(C3(C)CC3)=O)OCC2)=O)cc(F)c(C#N)c(F)c1 32763,CC1CN(C(=O)CCCF)CCC1CNC(c1cc(Cl)ccc1Cl)=O 32764,c1(CN(C(C2CC(CCNC(c3ccc[nH]3)=O)C2)=O)CC)cnc[nH]1 32765,C(CCCCCC(=O)NCC1CC(CO)CO1)NC(c1n(CC)nc(C)c1)=O 32766,c1(C(=O)NC(C2CCCN(C(=O)CCNC(=O)CO)C2)C)ncnc(O)c1F 32767,CC(CNC(=O)COC1CC=CC1)(C1CC1)NC(=O)Cc1cnoc1 32768,C1(C(C)C(=O)NCC(C2CC2)C2CC2)CCN(C(=O)COC2CCCOC2)C1 32769,N1(C(C(C)OCCC=C)=O)CC(CO)C2(C1)CN(C(c1ccc(CCC)s1)=O)C2 32770,C=Cc1ccc(C(N2CC(CN(C(=O)C(Cc3ccccc3)OC)C)C2)=O)cc1 32771,C1(CCC(=O)N(CC(C)N(C(CCCC)=O)C)C)CCCC(O)C1 32772,N1(C(=O)C2=CCCSC2)CCN(C(=O)COc2cccnc2)C2CCCCC2C1 32773,C=C(Br)CCC(=O)N1CCN(CCCNC(c2snnc2C)=O)CC1 32774,c1(C(=O)NCC2C(NC(c3cnn(C)n3)=O)CCC2)cc(Cl)cc(C(F)(F)F)n1 32775,N1(C(CCC)=O)CC2CCC(C1)C(NC(=O)C1=CC(C)(CC)C1)C2 32776,C1(N(CCNS(CC)(=O)=O)C(c2ccn(C)n2)=O)CC2CCC(C1)N2 32777,C1(NC(C2(OC)CCCCC2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)CC1C 32778,n1(CC)ccnc1C=CC(=O)NCCC1CN(C(C2CC(CC3CC3)C2)=O)C1 32779,S(=O)(=O)(c1cc(C)c(-c2ccccc2C#N)cc1C)NC(CC)CCN(C)C 32780,CC1=C(C(=O)NC2C3CC4C(C3)C24C(=O)Nc2cn(C)nc2Cl)SCCO1 32781,c1(C(N2C3C(NC(C4CC(=C)C4)=O)CC(CC3)C2)=O)ccc2cc(Cl)ccc2n1 32782,c1(C(=O)NCCN(C(=O)C2=CCCO2)CC)cccc2nccn12 32783,Cc1nnc(CCC(=O)NC2(CCNC(c3ccc(Cl)cc3)=O)CCC2)n1C 32784,C(=O)(CCC(C)(C)NC(=O)CCCn1cccn1)N(c1cccc(F)c1)CC 32785,N1(C(c2cn(CCC)nc2C)=O)CCC(C)(NC(c2n[nH]c(C)c2C)=O)CC1 32786,C(CCO)(C(F)(F)F)NC(c1c(CCNC(Cc2nc(C)[nH]n2)=O)n[nH]c1)=O 32787,CCC(O)C(C)(C)C(=O)NC1CC(NC(=O)C(C)(C)ONC(=O)OC(C)(C)C)C1 32788,c1(C(N2CC(N3CCC3)CC(C)C2)=O)ncc2cc(Br)ccc2n1 32789,N1(C(CC(CC)C2CC2)=O)CCC2C(NC(c3c(C)nn(CC)c3Cl)=O)CC12 32790,Cc1cc(Cl)ccc1C(N1CC(CNC(C2(n3cnnn3)CC2)=O)C2(CC2)C1)=O 32791,c1(C(=O)NCC23N(C(C(C)=C4CCC4)=O)CC(C2)C3)ccc(C)cc1N=[N+]=[N-] 32792,c1(C(=O)NCCCNC(c2c(C)ccc(OC)n2)=O)nccc2c1NCCC2 32793,c1(NC2(N(C(=O)CSC(F)F)C(c3ccccc3)=O)CCCCC2)ncc([N+](=O)[O-])cn1 32794,CC(C)(C)CC(=O)N(CCCNC(C12CCC(CC1)C2)=O)C1CC1.C1C(=O)N1 32795,c1(N(c2c(OC)c(F)ccc2)C(C2CC3CCCCN3C2)=O)ccnc2ccnn12 32796,c1(COC)nc(NCC(C)N(C)C(C)C)cc(N2CCC(C(C)CO)CC2)n1 32797,N1(C(N2CC3C(C(N(CCN(C)CCO)C)=O)(C3)C2)=O)C(=O)CCCC1=O 32798,c1(CCC(=O)N(CC(C)N(C(=O)CCC(F)F)C)C)ccccc1C(=O)N(C)C 32799,C1(C(N2CCC(O)(CN(C(c3c(C)cc(CC)o3)=O)C)C2)=O)CCCCCN1C 32800,CC1OCCCC1C(=O)N(C)CCN1CCN(C(=O)CC2OCCO2)CC1 32801,Cc1cc(=NC2CN(CC3CC3)C2)[nH]c(N2CCc3n[nH]cc3C2)n1 32802,CCC(CC)CC(=O)NCC(C1(O)CN(C(=O)CCF)C1)(C)C 32803,C(C(C)C)(C(O)C(=O)NCC=CC(=O)NCC1CCC(C)(C)CC1)OC 32804,C1(C(=O)NC2CN(CC)C(=O)C2)CCC(C)(C)N(C(=O)CN(C)C2CC2)C1 32805,N1(C(C=Cc2n(C)ccc2)=O)CCC2(CCCCN(C(C3C=CCC3)=O)C2)C1 32806,Cc1cc(N)cnc1C(=O)NCC(C)NC(c1cnsc1C)=O 32807,CC1CC(NC(c2cnc(-c3cccnc3)s2)=O)CN(C(=O)CC2CC=CC2)C1 32808,C(C)(C)(CCC(=O)NCCCCOC(C)C)NC(C(COCC)C)=O 32809,C1(CNC(C(C)OCC=C)=O)CCN(C(C2CC2c2cccc(Cl)c2)=O)CC1 32810,C1(NC(c2cnn(C(C)(C)C)n2)=O)CCC(C)(CNC(=O)C=Cc2ncc[nH]2)C1 32811,C12(CCNC(=O)C=Cc3cnc[nH]3)CCC1CN(C(c1cc3sccc3[nH]1)=O)C2 32812,N1(C(C(CC=C)C)=O)CCC2CN(C(c3ccccn3)=O)C(C)C12 32813,C(CCC(C(=O)N1CCN(C(C)C)CC1)NC(=O)CC(C)n1cccc1)OC 32814,C1(C(N2CC(N(C)C(c3cnn(C)c3)=O)C(C)(C)C2)=O)(OC)CCCCCCC1 32815,C1(C(=O)NC(C(C)C)CNC(=O)CC2CCN(C)C2=O)CC(=O)OC1(C)C 32816,C1(CNC(NCC(C)C)=NCC=CC2CC2)CSc2ccccc2O1 32817,CC1(C)OC2(CNC(C3(C4CCCO4)CCCO3)=O)CC1(NC(=O)CCF)C2 32818,n1(CCN(CCCC)CC)cc(C(O)CC)nn1 32819,N1(C(CS(CCOC)(=O)=O)=O)CCC2(CC1)CN(C(C1CC1OC)=O)CCO2 32820,C1(CC(C)(C)NC(C23CCC(CC2)NC3=O)=O)C(CN)C2CCC1(C)C2(C)C 32821,CCCC(CNC(=O)CCC1CCCCC1)NC(c1sncc1C)=O 32822,C1(NC(c2ccc(C)cc2C)=O)CN(C(=O)CC2CN(C)C2)C2(CCCC2)C1 32823,C1(NC(CNS(NC)(=O)=O)=O)CC2CCC1C(NC(c1ccnc(CO)c1)=O)C2 32824,c1(NC(C(C)S)=O)ccc2c(c1)CCN(C(c1cccn3nccc13)=O)C2 32825,c1(C(N(CCC)CCNC(=O)CN2CCOCC2)=O)ccc(O)cn1 32826,CCCC(C)(c1nnnn1CCCF)NC1CCC1(C)C 32827,C1(NC(C(n2c(C)cc(C)n2)C)=O)CC2CCC(C1)N2C(c1ncccc1C)=O 32828,c1(CC)oc(C)cc1C(=O)N(C(C)CC(=O)NCCC(F)F)C 32829,c1(C(=O)NC2CCCN(C(=O)CCCn3cccc3)C2)cc2nc(F)ccc2o1 32830,Cc1sc(=O)n(CC(N2CCC(NC(C3CCC(C)CC3)=O)C2)=O)c1C 32831,N1(C(=O)CCC(F)(F)F)CCC2CCN(C(c3ncn4c3CCC4)=O)C2C1 32832,c1(C(=O)NC(C)C(CO)NC(c2ccc[nH]2)=O)cccc(-c2cnco2)c1 32833,C(=O)(C1CCCc2nnn(C)c21)N1CCCN(C(c2c(C#C)c[nH]n2)=O)CC1 32834,N1(C(c2cc(C)nn2C)=O)CC2CCN(C(=O)CC3CCCCCCC3)CC2C1 32835,CC1(C)CCOC1C(=O)N(C1CCCN(C(=O)CCNC(=O)CO)C1)CCO 32836,c1(C(N(C(C)CNC(=O)CCCc2cncs2)C)=O)cc2c(O)ncnc2cn1 32837,Cc1cc(NC(=O)CC2C(NC(C3C(C)(C)C3(F)F)=O)CC2O)cc(CO)c1 32838,C(=O)(C1Cc2ccc(C)cc21)N1CCN(C(c2cc(CC)c(C)s2)=O)CC(O)C1 32839,N1(C(C(C=C)O)=O)CC2(CCN(C(c3c(C)oc(C)c3C)=O)CC2)C1 32840,N1(C(CN(C)CC)=O)C2CCC1CC(CNC(c1cnn(C)c1C(C)C)=O)C2 32841,C(=O)(C(C(C)(C)C)n1cc(-c2n[nH]c(C)c2-c2nn[nH]n2)nn1)NC 32842,C(=O)(C(F)CC(C)C)N(C1CCN(C(=O)CN(S(=O)(=O)CC)C)CC1)CCC 32843,C=CC(CC)CC(=O)N1CCC(C)C(NC(=O)C=Cc2cnc(OC)nc2)C1 32844,C1(NC(CCn2ccc(C)n2)=O)C2CC3CN(C(C4OCCCO4)=O)C1C3C2 32845,C1(C(N2CC(NC(=O)C=C3CCCC3)C2)=O)CC12CCCc1ccccc12 32846,C1(NC(C2CC(OCC)C2)=O)CC(NC(C2(C(C)(C)C)CCCC2)=O)C12CCC2 32847,C(=O)(CC(O)CCSC)NC1CCN(C(c2ccc(CC)nc2)=O)C1 32848,C12(NC(c3nc(C(C)(C)C)oc3)=O)CCCN(C(=O)C3=CCC3)CC1C2 32849,c1(C(C)C(=O)N(CC(=O)N(C2CCCCO2)CC2CC2)C)cccc(COC2CC2)c1 32850,c1(N(CC(c2ccccc2)(C)C)C)c(CNC(C)C(=O)OC)cccc1F 32851,c1(-c2n(C)ncc2)cccc(C(=O)NC2CC(NC(=O)C=CC(F)F)CC2O)c1 32852,CC1(NC(=O)CN(C)C2CC2)CN(C(C2CC(n3cnnc3)C2)=O)C1 32853,N1(C(=O)NCC2CC(N)(CC)C2)CCC(OCCO)CC1 32854,c1(C(N2C(C(=O)NCC3COCCO3)CCC2)=O)cc([N+](=O)[O-])cs1 32855,c1(OCC(=O)N(C2CCN(C(C(C)=CC3CC3)=O)C2)CCO)c(C)cccc1Cl 32856,C1(C)(C(=O)NCCCN(C(C2CCc3ncnn3C2)=O)CC)CC(C2CC2)=NO1 32857,N1(C(C(C)(C)OCC)=O)CCN(C(c2c[nH]cc2CC)=O)CC(O)C1 32858,O=S(=O)(c1cccnc1NCC1CC2(C1)OCCO2)N1CCCC1CF 32859,c1(C(N2CC(C)N(C(c3ccc(N(C)C)nc3)=O)CC2)=O)ccn2ccnc2n1 32860,Cc1onc(-c2cccc(F)c2)c1C(=O)NC(C)CN(C)C(c1coc(Cl)n1)=O 32861,c1(NC(C2C(CNC(Cc3n(C)ccc3)=O)C2)=O)cnc2[nH]cnc2c1 32862,c1(CNC(=O)NC(c2cn(C)nn2)c2cccs2)cc(Cl)ccn1 32863,c1(-c2cn(CC3N(C(CC(CC)C(F)F)=O)CC3)nn2)ccc2nccnc2c1 32864,C(=O)(CCS(=O)(=O)c1ccc(OC)cc1)NCCNC(C(CCCC)(C)F)=O 32865,c1(C(C(=O)NC)N(CC)Cc2cccc3ccsc23)ccc2c(c1)CCOC2 32866,c1(C(N(C(CNC)C)C)=O)cc(F)c(O)c(Cl)c1.Cc1cc(CC=O)on1 32867,N1(C(Cc2cc(C)no2)=O)CCCC(C2CC2NC(c2cc(C(N)=O)cs2)=O)C1 32868,c1(C(=O)NCC2CN(C(C(C)NC(C)=O)=O)CC2C)cccc2c1CCC2 32869,N1(C(CC23C(C)(C)C(CC2)CC3)=O)CCCC(C2(NC(=O)C(O)C3CC3)CC2)C1 32870,c1(C(N2CC(OCCNC(C3C(C)(C)OCC3)=O)C2)=O)n[nH]c2ccc(Cl)cc12 32871,c1(C(N(CCCCN(C(C(COC)OC)=O)C)C)=O)ccc2c(c1)C(C)C(C)O2 32872,C1(C(N2C(C(=O)NC(CCCC)C)CC3CC32)=O)CC2(C1)CC(O)C2 32873,C1(C(N2CCC(N(C(=O)CN3CSCC3=O)C)CC2)=O)C(C2CC2)C1(F)F 32874,c1(NC(C2N(C(c3c(C)c[nH]c3)=O)CC(C)C2)=O)ccc2c(c1)ncn2C 32875,CCC(C(F)F)NC(=O)Nc1csc(CNC(=O)OC(C)(C)C)c1 32876,CC(C)C(C)C(CNC(C1CCSCC1)=O)NC(c1cc(=O)n(C)o1)=O 32877,N1(C(CC2ON=C(C)C2)=O)C(CC(=O)NC(C)(C)CC(C)(C)O)C2CCCC12 32878,C(=O)(C1=CC2(CCOC2)C1)NCC1(NC(c2c(C)ncnc2)=O)CCCCCC1 32879,Fc1ccc(Cl)c2[nH]cc(-c3nc(-c4cccnc4)nn3NCC3CCOC3)c12 32880,N1(c2c(C)c(NCCCC(F)F)ncn2)CCOc2cc(Cl)ccc2C1 32881,c1(C(=O)NCCC(C)NC(=O)Cc2cncs2)cccc(N)c1 32882,C1(C(=O)NCC(N(C(c2scc(C)c2Cl)=O)C)C2CC2)CCn2nnnc2C1 32883,C1(C(N2CCC(CCCC)C2)=O)C2CC1N(C(c1cc(C(C)C)no1)=O)C2 32884,CC(=O)C(C)(C)CC(=O)NC(C1CN(C(C2CS(=O)(=O)C2)=O)C1)C 32885,C1(CNC(c2n(CCOC)ncc2)=O)CC2CC2N1C(C1CCCOCC1)=O 32886,C1(CC=C)(NC(=O)CC(C)CF)CCN(C(=O)C=Cc2ccccc2)CC1 32887,c1(SCCNC(=O)CO)nnnn1C1CCCCC1 32888,C1(NC(c2c(C)noc2N)=O)CC2CC(C1)N(C(=O)CP(C)(C)=O)C2 32889,N1(C(C2C(C=C)C2)=O)CCC2(CC1)CCN(C(C1CCCC1(C)C)=O)CC2 32890,C(=O)(C(C(C)C1CCOC1)N1CCC2CC2C1)N(CC(C)C)C(=O)OC(C)(C)C 32891,C(=O)(CCCN(C)N=O)NC1(CC)CCCN(C(=O)CCc2ccc(F)cc2)C1 32892,N1(C(=O)NCC(=O)NC2CC2)CC2CC1CN2C(c1csc(Br)n1)=O 32893,c1(OCCC(N2CCC(OCCNC(=O)C3=CCC3)C2)=O)ccc(Cl)cc1Cl 32894,CC1(NC(=O)COCCc2cccs2)CC(NC(=O)C=CCN2CCCC2)C1 32895,C#CCC(CC(=O)NCCOC1(C)CCC1)NC(C1CC12CCCC2)=O 32896,CC(F)(F)C(F)C(=O)NCc1ccc(C(=O)NOCCCCCC2CC2)s1 32897,Cc1ccc(C(C)C)c(NC(=O)CC(C)C)c1.C123CC(CO1)(C2)C(=O)NC3 32898,C1(NC(C(=O)NCC2CC2)=O)C2CC(CN(C(C3CC4C=CC3O4)=O)C2)C1CO 32899,C1(CNC(C=CC(=O)OCC)=O)CC(C(=O)N2CCC(CO)(OC)C2)=NO1 32900,C=CCC(CNC(C1CCCO1)=O)C(=O)NC1(COC)CCCC1 32901,c1(C(=O)NCC2CC(C)(C)N(C(C3CCC(=O)NC3)=O)C2)nccc2n[nH]cc12 32902,C1(CC=C)CN(C(C2CN(C)C2)=O)CCCO1.C12(CCC1CC)C(=O)N2 32903,C(=O)(C(C)CCCc1cccs1)N1CC(=C(CNC(CCC)=O)F)C1.OC 32904,c1(NCC(N2CCC(NC(C(C)NC(C)=O)=O)C2)=O)ccc(C(F)(F)F)cc1 32905,N1(C(c2c(C)nc3sccn32)=O)CCC2(CCC(NC(=O)C3=COCCC3)C2)C1 32906,N1(C(c2n(CC)nnc2)=O)CCN(C(=O)CCc2ccc(Cl)s2)CC1C 32907,c1(C(N2CCCC(c3nnc(C)o3)C2)C(=O)NC(C)C)sc(C#N)cc1C 32908,C1(C)(COC)CC(NC(c2c(C)ccn2C)=O)CN1C(c1cc(CO)[nH]n1)=O 32909,N1(C(CN(c2ccccc2)CC)=O)C(C)CC2CN(C(C3CCNC3=O)=O)CC12 32910,C1(OC)CC2(C1)CN(C(c1csc(CNC(C3(CF)CC3)=O)c1)=O)C2 32911,c1(C(=O)NC(CCNC(c2ccn(CC)n2)=O)C)ccc(C2CNC(=O)C2)cc1 32912,CCC(C)C(C(=O)N1CCC(O)CC1C(=O)NC(CO)C(C)C)N(C)C 32913,C(CC1=CCN(C(c2cc(N)nc(Br)c2)=O)CC1)NC(C1C(=C)C1)=O 32914,C(CC(O)CC(=O)N1CC2C(NC(c3[nH]nnc3C3CC3)=O)C2C1)SC 32915,N1(C(c2ccccc2)=O)CCCC(C2CCCN(C(C3CC(O)C3)=O)C2)C1 32916,N1(C(COCC)=O)CCCC(C)(CNC(=O)C2=CCCC2C)C1 32917,C=C(C)CCC(=O)NCC(C1CCCCC1)NC(=O)COCc1cccnc1 32918,c1(CNCC(C2(OC)CCCC2)(F)F)ncc(Br)cc1Br 32919,c1(-n2cc(C(C)NC(=O)CC3CC4(CC4)C3)nn2)ccc(Cl)c(F)c1 32920,C1(C(=O)NCC(=O)NCC#C)CC1C1CN(C(C2CC(C(C)C)C2)=O)C1 32921,CC1=CN2C(C(=O)NCCCCN(C)C(C3CC4CC4C3)=O)(C=C1)CC2 32922,N1(C(C(OC)OC)=O)CC2CC(NC(c3conc3C3CCC3)=O)CC1C2 32923,Cc1ccc(C(=O)NC(C)CCNC(=O)COCC2CCCO2)c(N)c1F 32924,c1(C(N2CCC(NC(CCS(=O)(=O)NC)=O)C(F)C2)=O)cnc2c(c1)CCCO2 32925,C1(OC)CCN(C(c2coc(-c3ccsc3)c2)=O)CC1C.C12CC(C1)C2CC 32926,c1(CCC)ccc(C(=O)NCC(C)N(C(=O)CSCCC#N)C)cc1.N1(C)CCCC1 32927,C(=O)(C(O)C(F)(F)F)NCC1CC(C)N1C(=O)CC(C)(C)C 32928,CCC(Cc1ccccc1)C(=O)N1CC(C)(NC(=O)CCC(=O)NC)C1 32929,N1(C(C(=O)NCc2ccc(F)cc2)C2CC2Cl)CCCC2CC(O)CCC12 32930,Cc1nc(O)ccc1C(N1CCC(C)C1C(=O)Nc1cnn(CCF)c1)=O 32931,C1(NC(C(C=C)O)=O)CCN(C(c2c(OC)noc2C2CC2)=O)CC12CCC2 32932,c1(OC)ccc(C(N2CCCC2C(C)(C)CNC(C2CN(C)CC2O)=O)=O)nn1 32933,CCCC(F)C(=O)NCCOCCCN(C)C(C1CCC1C#N)=O 32934,C(C(=O)NCC1CCN(C(C2CCOCC2(C)C)=O)C1)(c1ccccc1)=C(C)C 32935,CC(C)CC(CC(C)C)C(=O)NCCC(C)N(C(=O)CCc1ncc(F)cn1)C 32936,CN1CC=C(CCNC(C2CCCCC2(C)NC(=O)C2=NOC(C)(C)C2)=O)CC1 32937,c1(CN2C3CC(C(=O)Nc4c(CC)ncs4)CC2CC3)nc2ccc(C)cc2[nH]1 32938,C1(CNC(C(C)(C)SC)=O)CN(C)CCN1C(c1cc(Cl)sc1Cl)=O 32939,Fc1conc1COC(C1CCCC1c1nc[nH]n1)=O 32940,CC(F)(F)C(C)(C)CC(=O)N1CC(NC(C2CC(O)C2)=O)CC12CCOC2 32941,C(=O)(C1Cc2ccccc21)NC(CCC(C)C)C(=O)NC(CO)C(=O)N(C)C 32942,c1(C(N(CCC(=O)N(CC)CC)CCC)=O)cn(C2CC2)nc1C 32943,N1(C(CC2CCC(=O)C2)=O)CC2(CCC(CNC(c3ccoc3Br)=O)O2)C1 32944,C1(C(=O)NCC2(NC(c3cnc(-c4ccco4)s3)=O)CC2)CCC2(CC2)C1 32945,C1(O)(CN(C(C2CCN(C)C2)=O)C)CCN(C(=O)CCc2cnn[nH]2)CC1 32946,c1(CC2N(CC(O)Cn3ccc(C(F)(F)F)n3)CCC2)cccc2[nH]ccc12 32947,C1(C)(COC)CC(NC(C2CN(C)C2)=O)CN1C(=O)CCc1nncs1 32948,CCCC(CCC)CC(=O)NC(C1CC=CCC1)C(=O)N(CCCCCO)C 32949,c1(C(=O)NC2(CNC(C3C(CC)C3)=O)CC2)cncc(Cl)c1C 32950,N1(C(c2c(CC)noc2)=O)CC2CC(C)N(C(c3cn(C)nc3Br)=O)C2C1 32951,c1(OC)cc(F)cc(C=CC(N2CCCC(C)(C)C2CNC(=O)C(C)SC)=O)c1 32952,c1(C(N2CC3(CC(NC(C4(F)CC4)=O)C3)C2)=O)ccc2nc(O)oc2c1 32953,C#Cc1cc(F)c(CN2CCN(C)C(CO)C2)c(F)c1 32954,N1(C(c2c(SC)n(C)nc2)=O)CC2CCCC2(CNC(=O)Cc2cc[nH]c2)C1 32955,C1(OCC)CC2(CCN(C(=O)CC=CC(C)(C)C)C2)C1.C12C(C1(C)C)NC2=O 32956,c1(N2CCCC(NC(c3cccc(C(C)(C)C)n3)=O)C2)ccnc2ncnn12 32957,CC(C)(Cc1ccccc1)C(=O)N1CCCC1NC(c1c[nH]ccc1=O)=O 32958,C1(C)(CNC(CN(C)CC)=O)CCCN1C(=O)Cc1cc(C)no1 32959,C(=O)(N=c1c(Cl)c[nH]cc1Br)C1C=CC(NC(c2c(C)noc2)=O)C1 32960,C(=O)(CCCCN=[N+]=[N-])NCC=C(C(N1CCC(C(=O)OC)CC1)=O)C 32961,Cc1cc(C(=O)NC2C3CC2N(C(=O)C(C)OCc2ccncc2)C3)cc(C)n1 32962,N1(C(c2ccc(CC)cc2O)=O)CCC2(CC(NC(=O)C(C)OCOC)C2)C1 32963,Cn1nncc1CC(=O)N(CCCNC(=O)C=CCOCC(F)(F)F)CCO 32964,c1(C(N2CCC(CNC(C3C(OCC)C3)=O)C2)=O)ccc(-c2ccc(Cl)s2)cn1 32965,C1(NC(c2ccsn2)=O)C2CC3C1C3C2C(N1CC(n2cccn2)C1)=O 32966,N1(C(C2CN(C(Cc3nc(C)sc3)=O)C2)=O)CCN(c2ccc(F)cc2)CC1 32967,C(=O)(C(O)C(F)(F)F)N1CC(CC(N2C(COC)COCC2)=O)C1 32968,c1(C(=O)NCCOCCCNC(CC2C(C)C2)=O)ccc(OCF)nn1 32969,c1(N(C)CCn2cccn2)ccnc(NCC2CC2(F)F)n1 32970,C1(N(C(C2(CC)CCC2)=O)C)CC2CCC(C1)N2C(c1occ2c1CCC2)=O 32971,C1(OC)CC(CO)(NC(=O)CC2C=CC(NC(=O)CCCC3CC3C)C2)C1 32972,C=CCCCCCCCCC(C(=O)NC1CC1)N1CCCC(CCCO)C1 32973,N1(Cc2ccc(C(=O)OC)cc2C(F)(F)F)CCc2c(C)cccc2C1C(=O)O 32974,N1(CC)CCC(C(=O)NCC(c2ccccc2)N(C(=O)CC2CC(=O)C2)C)C1 32975,c1(C(C(=O)NCCCC)N(C)C)cn(CCCN2CCC(C(=O)N(C)C)C2)nn1 32976,c1(N2CCC(CNC(C(C)CN3CCOCC3)=O)C2)cccc(O)n1 32977,S(=O)(=O)(c1ccc(Br)cc1)NCC(=O)NCCNC(c1cccc(CO)c1)=O 32978,N1(C(CCC(=O)OCC)=O)CC(O)C(O)C1CNC(c1ccc(C)c(CO)c1)=O 32979,N1(C(c2cnc(Br)s2)C(=O)NCCSC)CCCC(n2cc(C)cn2)C1 32980,N1(C(CCCCSC)=O)CC(NC(c2nc(C3CC3)ncc2Cl)=O)C(C2CC2)C1 32981,c1(CC(=O)NC(CC)CN(C(=O)C(C2CC2)C2CC2)C)cc(F)ccc1C 32982,N1(C(c2ccc(CSC)cc2)=O)CCCN(C(=O)COC(F)(F)F)C(CO)C1 32983,N1(C(c2ccn(C(C)(C)C)n2)=O)CCOC(CCNC(c2nocc2Cl)=O)C1 32984,C(C(C(C)(C)C)NC(C1(C)CCCO1)=O)NC(=O)Cc1csc(C(F)(F)F)n1 32985,CCC(C)(C)CCNC(=O)C=CC(C)(C)NC(=O)C(C)C(F)F 32986,c1(CC(=O)OC)ccc(CNC(=NCc2cnccn2)NC2CCCCC2)cc1 32987,Cc1c(CCNC(CC(C)C)c2nnnn2C2CCCCC2)cccc1Br 32988,N1(C(C(c2cc(C)c(C)s2)NC(=O)OC(C)(C)C)=O)CCCC(C2(C)CC2)C1 32989,C(CCF)(C(=O)NCC1C(C)C1(F)F)NC(c1cc(C)[nH]c1)=O 32990,C(=O)(C1=C2CCN=C2NC=C1)NC(CCCOC)c1cccnc1 32991,C1(C(N2CCC(=CCNC(C(CCC)NC(N)=O)=O)CC2)=O)CCCS(=O)(=O)C1 32992,C1(COC)CN(C(c2cc(C#N)[nH]c2C)=O)CCN1C(=O)C1=C(Cl)CCC1 32993,C1(OC)CCn2cc(C(=O)NCC3CCCCN3C(=O)C(CO)N(C)C)nc2C1 32994,C(c1cncnc1O)=CC(N1CCC(C(C)NC(=O)CC(F)(F)F)C1)=O 32995,N1(C(Cc2cc(C)[nH]n2)=O)CCOCC(C)(CNC(C2CCC2C(C)(C)C)=O)C1 32996,N1(C(c2n(C)cnc2)=O)CCOC(C2CN(C(C3CC=CCC3)=O)C2)C1 32997,C1(CC)CCC(C(=O)N(CC(C)O)CCN(C(=O)CCc2csc(C)n2)C(C)C)O1 32998,N1(C(C(C)N(C(C(CCCC#C)C)=O)CC)=O)CC2CCC1C(O)C2O 32999,c1(C(N(CCCCNC(C(CCC)O)=O)C)=O)cc(F)cc2c1NCCC2 33000,C1(C(=O)NCC(CN(C)C(C2CCC(=O)C2)=O)(C)C)CCCC1P(C)(C)=O 33001,c1(C(=O)NCCN(CCOC)C(c2nnn(C)c2C)=O)cc2ncn(C)c2cn1 33002,c1(CN2CCC(N(C(=O)CCCN3CCCCC3)CC)C2)ccc2nonc2c1 33003,Cc1cc(C(=O)NCC2CCC(NC(=O)CCCCNC(N)=O)C2)c(C)cn1 33004,Cc1nn(CCC#N)c(C)c1C(=O)NCCCc1cn(CCCS(N)(=O)=O)nn1 33005,CC(C(C)(C)C)=CC(=O)NCCCOCCC(=O)NCC1=CCCC1 33006,c1(C(=O)NCC(C)NC(C(c2cccc(OC)c2)O)=O)cc2nc(F)ccc2o1 33007,S(=O)(=O)(c1cccc(C#N)c1)N1C2CC(NC(c3cn(C)nc3)=O)CC1CC2 33008,[N-]=[N+]=NC1CCCN(C(c2csc3ccccc23)=O)C1 33009,C(c1cnc2ccccc2n1)=CC(=O)NC1C2CN(C(CC(C)(C)O)=O)C1CC2 33010,c1(NC(N(CC(C)C(=O)NC)CCC)=O)cc(Cl)c(Cl)cc1OC 33011,Cc1cc(C(=O)N(C2CN(C(=O)CN(C)C)CC2(C)C)C)c2nc(C)n(C)c2n1 33012,C1(C(=O)NC2COCC2CNC(C2CCCCC2(C)C)=O)(CC)CCC(O)CC1 33013,S(=O)(=O)(c1ccc(Br)cc1NC(c1ccccc1)CO)N(C)CC1CN(C)C1 33014,C(c1cccc(F)c1)=CCC(=O)NC1COCCC1NC(c1cccnc1)=O 33015,c1(N(CC(c2ccccc2)(C)F)C)ncnc(NCc2nnc(C)s2)c1C 33016,Cc1cc(=NCC2CCCN(C(C3(F)CC4(CCC4)C3)=O)C2)[nH]c(C2CC2)n1 33017,N1(C(CC2CCC(NC(COC3(C#C)COC3)=O)CC2)=O)CCC(O)C(C)C1 33018,N1(C(C(CC=C)C)=O)CC(NC(c2cccc(C(F)F)n2)=O)C2(CCOCC2)C1 33019,c1(C(N2CC(C=C)C(NC(c3[nH]nnc3C)=O)C2)=O)nn(C)c2c1C(O)CCC2 33020,N1(C(c2cnc(C)n2C)=O)CCn2ncc(CNC(C3CCS(=O)CC3)=O)c2C1 33021,N1(C(C2C(C)CC(=O)N2)=O)CCC2(C1)CN(C(=O)CC1CCCC(F)(F)C1)C2 33022,c1(CNC(=NC)N(C)Cc2conc2CC)cccc2c1OCCO2 33023,c1(CC)ccc(NC(=O)C(CC2CCCC2)NC(C2CCC(COC)O2)=O)cc1 33024,CC(CC(C)(C)C)C(=O)N1CC2(CCN(C(C3(CN(C)C)CCCC3)=O)C2)C1 33025,C1(C(=O)NCC(C(C)(C)C)NC(=O)C=Cc2ccc[nH]2)CC2CCC1CC2 33026,n1(CCCC)ncc(C(=O)NCC2(Nc3nnc(C(C)(C)C)s3)CC2)c1C 33027,N1(C(CN(C)C2CC2)=O)CCC(C2CCCCN2C(=O)COCC2CCCO2)CC1 33028,C(=O)(C(C)(O)C(F)(F)F)N1CC(C(C)C)C(C(N2CCC(C)(C)C2C)=O)C1 33029,C(=O)(C(C)CC(F)(F)F)NCC1CN(C(c2c(C(C)C)ncs2)=O)CC1(F)F 33030,N1(C(CC2N(C)CCC2)=O)CCC(CC(N)=O)(NC(=O)Cc2nccn2C)CC1 33031,CCC(CC)CCCC(=O)NC(C1CCCC1)CNC(C1CC(=O)N(OC)C1)=O 33032,N1(C(C(CC(C)C)=O)=O)CCc2nc(O)cc(C(=O)NCCc3nccs3)c2C1 33033,C(=O)(CCCS(N)(=O)=O)NCC1CC(NC(C=Cc2ncc(C)[nH]2)=O)CC1O 33034,N1(C(C2(Nc3ccccc3)CC2)=O)CCOCC(NC(c2ccsc2)=O)C1 33035,c1(C(=O)NCCC(C)NC(c2c(OC)cncc2)=O)cc(Br)c(C)nc1O 33036,C(=O)(C(CC(C)(C)C)OC)NC1C(OC)CN(C(=O)CSC2CC2)C1 33037,c1(C(N2CCC(NC(C3CN4CCN3CC4)=O)C2)=O)cc(F)c(F)cc1F 33038,Cc1nc2sccn2c1C(N1CCC(C)(CNC(C2CC3CC3C2)=O)C1)=O 33039,C1(CCNC(CC(C)(C)C)=O)CN(C(C2CC2c2cccc(F)c2)=O)CCCO1 33040,N1(C(C)=O)CC2OC(=O)N(C3CCN(C(c4cc(O)n(C)n4)=O)CC3)C2C1 33041,C1(NC(=O)C2=CCCC2)C2CC3C1C3C2C(=O)NCc1cccc(F)c1O 33042,C(=O)(C(C(C)C)n1cc(Br)cn1)N(CCNC(=O)CSC(C)(C)C)CC 33043,CC(=NOCC#N)C(=O)N1CCN(CCNC(c2cc(C)ncn2)=O)CC1 33044,N1(C(CCC)=O)CC(OC)CC1(C)CNC(c1ccc(C)nc1O)=O 33045,C1(CNC(c2c(CC)nco2)=O)CN(C(=O)Cc2c(C)nn(C)c2Cl)CCN1C 33046,C1(O)(C(C)NC(=O)CCN(C)C2CC2)CCN(C(SC(F)(F)F)=O)CC1 33047,C1(C(c2nnnn2C2CCC2)NCCc2nnc(C(C)C)s2)(OC)CCCOC1 33048,C(C(C)(O)CC(=O)N1CC2(CC2)CC1CC(=O)N(CC(C)CO)C)OC 33049,N1(C(Cc2nc(C)sc2)=O)CCC(C)C(NC(=O)CCNC(=O)C(C)(C)C)C1C 33050,c1(C(N(CCC)CCNC(=O)CN(C)S(N)(=O)=O)=O)cnc2c(c1)CCCO2 33051,c1(C(=O)NCC(CN(C(CCOCC)=O)C)C)cc(C)c2nc(C)nn2c1 33052,C#CC1(C)CCCN(C(=O)C(=O)NC(c2cccc(C(F)(F)F)c2)COC)C1 33053,N1(C(C2CC(OC)C2)=O)CC(NC(c2cc(C)cc(O)n2)=O)C2(CCC2)C1 33054,N1(C(c2n(CC)ncc2)=O)CC2CC(C1)CN(C(=O)COC1CC1)C2 33055,C1(CC(=O)N(CC(C)O)CCNC(C=C(CCC)C)=O)CCCC(F)(F)C1 33056,C1(N(C(CCc2c(C)n[nH]c2C)=O)C)CCCCN(C(C2CCOC2)=O)C1 33057,C1(COC)(NC(c2cnn(C)c2F)=O)CCN(C(=O)CC2CCCO2)CC1 33058,N1(S(=O)(=O)C2CC2)CC2CCC(C1)N2Cc1ncccc1F 33059,CC(C)CCC(C(=O)NC1CCCC1CN(C)C)NC(=O)C=Cc1nccs1 33060,Cc1cc(Cl)c(C(=O)NC(C)Cn2cc(CNC(=O)C(C)O)nn2)c(Cl)c1 33061,CCCC(C)CN(C(=O)C(C)N(C(=O)CC(C)n1cccc1)CCC)C 33062,C1(C(=O)NCCCN(C)C(C23CCCC2C3)=O)CCc2ncccc2C1 33063,c1(C(=O)NCC=C2CCN(C(C3(Cl)C(C)(C)C3)=O)CC2)cc2c(nn1)CCC2 33064,c1(C(N2CC(CNC(C(C)(C)C3CCC3)=O)C3C2C3)=O)cccc2c1CCC2=O 33065,C1(C(=O)NCCN(CCC)C(c2c[nH]c(=N)s2)=O)COCCN1CC(F)F 33066,C1(CNC(=O)Cn2cncn2)CN(C(C2CC3CC(=O)C2O3)=O)CC1(F)F 33067,c1(C(N(CCNC(=O)C(C)OCC(F)(F)F)CC)=O)cn2nc(C)cc2[nH]c1=O 33068,c1(CC)ccc(C(=O)NC(C)C(C)NC(c2ccc(C3CC3)nc2)=O)cc1F 33069,Cc1cc(C(N2CCC3(CC3C(=O)NCCCC3CCCCC3)C2)=O)nc(C)n1 33070,CN1N=C(C(=O)N2CC3CCOCC3(NC(=O)CCc3cnc[nH]3)C2)CCC1=O 33071,C(=O)(CCC(F)(F)F)NC(CN1CCN(C(c2ccnc(C(C)C)n2)=O)CC1)C 33072,N1(C(c2cc(C(C)=O)oc2C)=O)CCCN(C(C2(N(C)C)CCCCC2)=O)CC1C 33073,N1(C(=O)Cn2ccc(C(F)F)n2)CC2CN(C(C3CC3(F)F)=O)CC2C1 33074,Cn1cnc2c1CCCC2C(=O)NC1CCN(C(c2nc(Cl)sc2Cl)=O)CC1F 33075,C1(NC(C(C)NC(=O)CN2CCCC2=O)=O)CN(C)NC1=O 33076,c1(C=O)cccc(S(=O)(=O)C(F)F)c1.CS(=O)(=O)c1ccc(N2CCC2)nc1 33077,C1(CCNC(c2cc(C)nnc2)=O)CN(C(C2C(C)(C)OC2(C)C)=O)CC(C)O1 33078,C(CC(C(C)C)NC(=O)CCc1ccc(Cl)nc1)N(C(c1c(CC)ccs1)=O)C 33079,c1(C(C)=O)cc(Br)ccc1NC(c1cccs1)=O.c12ccc([nH]1)CCC(=O)NC2 33080,N1(CC2CC2)CC2CC1CN2Cc1ccc(OC(F)F)c(NC(=O)C(F)(F)F)c1 33081,C(=O)(C(C(C)C)NC=O)N(C1CCN(C(=O)C(c2ccccc2)SC)CC1)CC 33082,c1(C(=O)NCC2C(NC(C(C)OCC=C)=O)CC2)c[nH]c2c(C#N)cccc12 33083,N1(CC(=O)NC(CC)(C)CNC(c2cn(C(C)C)nn2)=O)C(=O)CC(C)(C)C1=O 33084,c1(C(=O)OC)cc(C(N2CC(N(C(=O)C3=C(C)CCC3)C)C(F)C2)=O)cc(F)c1 33085,Nc1cc(Cl)ccc1C(=O)NCC1CC(O)CN1C(=O)CC1CC2(CC2)CO1 33086,CCCCC(O)C(=O)NCCCC(CCC)NC(c1cc(CCC)n(C)n1)=O 33087,c1(C(C(=O)NC2C(NC(c3cn(CCC)nc3)=O)CC2)C)ccc(C#N)cc1 33088,c1(CN(C)Cc2nc(CCC)sc2)cccc(I)c1 33089,C1(OC)CN(C(c2ncncc2Cl)=O)CC1NC(c1ccc(OC(F)F)cn1)=O 33090,Nc1c(F)ccc(F)c1C(N1CCCOC(CNC(C2CC2C2CCC2)=O)C1)=O 33091,c1(CC2(CC(=O)NCC3CN(C(Cc4nnc(C)o4)=O)C3)CC2)ccc(F)cc1 33092,Cc1nc(N(C(C)CCNC(C2(C3CCCO3)CC2)=O)C)[nH]c(=N)n1 33093,C1(NC(C)=O)CCC(C(=O)NCCN2CCCC2=O)OC1 33094,Cn1nc(-c2cn(CC3CCN(C(=O)C(Br)Br)C3)nn2)cc1N 33095,c1(N2CCC3(CC(NC(C(CC)C)=O)C3)C2)ncnc2ccc(S(C)(=O)=O)cc12 33096,CC1(CNC(c2cc(C(F)F)no2)=O)CCN(C(C23CC(O)C2C3)=O)CC1 33097,c1(CC(=O)NC(C)CNC(=O)Cc2ccoc2)csc(CS(C)(=O)=O)n1 33098,c1(-c2nc(C(C)SCC)nn2CC)cnn2c1CC(C)CC2 33099,c1(CCC(N2CCC(C)(CNC(C(C)OCC#C)=O)C2)=O)c(O)nc(=N)[nH]c1C 33100,c1(N(C)C)ccc(C(=O)NC2(CCCNC(=O)CC(Cl)Cl)CC2)nc1 33101,C1(NC(C(N2CCNC2=O)C)=O)C2CC1N(C(C1CCSC1)=O)C2 33102,C1(NC(CCCC#CC)=O)CN(C(c2ccc(CC)[nH]2)=O)CC2(CCOCC2)C1 33103,C(c1cccc(F)c1)=C(C(=O)NC1C=CCN(C(c2c(CC)onc2C)=O)C1)F 33104,Cc1cccc(C(O)C(N2CCOC(CN(C(=O)Cc3nnc(C)s3)C)C2)=O)c1 33105,N1(C(C(C)NC(C23CC(CN(C)C)(CO2)C3)=O)=O)CCC(O)(CO)C1 33106,C1(CNC(C(C)OC(C)=O)=O)CCC(C(=O)N(C2CC3CC3C2)C)CC1 33107,C1(C(=O)NCCCC2OCCN(C(C(C)(C)N(C)C)=O)C2)CCCCC12CCC2 33108,C(CC(O)CC(=O)NCCCN(C(=O)CCCC(N)=O)Cc1ccccc1)SC 33109,c1(CC(C)C)cc(C(=O)NCC(C)NC(=O)CCc2cccnc2F)cc(O)n1 33110,c1(C(=O)NCCN(C(c2csc(C(=O)OC)c2)=O)CC)ccc(CC(C)C)nc1 33111,CCCCC(C(=O)N1CCCOC(CNC(=O)CCc2scnc2C)C1)N(C)C 33112,Cc1ccc(C(N2CCC(N(C(=O)C(O)Cc3ccccn3)C)C2)=O)cc1 33113,Cc1scc(CNC(=O)C(C2CC2)NC(=O)C(C)NC=O)c1C 33114,c1(N2CCC(CCC)(CO)C2)nc(=NCC(C)(C)N2CCCC2)[nH]c2c1CSC2 33115,C1(Cn2cc(C(C(C)(C)C)O)nn2)CCCN(C(=O)C(c2cscn2)N(C)C)C1 33116,c1(OC)cccc2c1OCCC2NS(=O)(=O)c1c(Br)cc(C(=O)O)cc1Br 33117,c1(OC)ncccc1C(=O)NCCCC(=O)NC(C)Cc1cnccn1 33118,N(C(=NC(C)C)N1CCC(F)C1)Cc1nn(CC)nc1C 33119,N1(C(c2c(OC)cc(C)cn2)=O)CC(NC(=O)C2=CCCC2C)C(N=[N+]=[N-])C1 33120,Brc1c(SCCCCc2ccc(Nc3ccc(Br)cc3)nc2)cc(Br)c2ncccc12 33121,C(=O)(C#CC1CCCOC1)NC1CC2CN(C(C=Cc3ccc(C)o3)=O)C(C1)C2 33122,c1(C(N(C)CC2CCN(C(=O)Cc3cncc(F)c3)C2)=O)cnc(N)c(N)c1 33123,Cc1ccc(C(=O)N(C)CC2CCCN2C(=O)CC2CC(CF)C2)cc1N 33124,c1(C(N2CCC(O)(C(C)NC(=O)CN3CCC(O)CC3)C2)=O)ccc2c(c1)CC2 33125,C#CCCC(C(=O)NC1(CC)CC(C)(C)C1)NC(C1CC2(C1)CC(C)C2)=O 33126,N1(C(C2CC(=O)N2)=O)Cc2ccc(CNC(c3ccc4nn[nH]c4n3)=O)cc2C1 33127,c1(C(=O)NCC2N(C(c3c(C)con3)=O)CC(O)C2)ccc2nc[nH]c2n1 33128,N1(C(C2CCC(CC)C2)=O)CCCN(C(c2cnn(CC(C)C)c2)=O)CCC1 33129,N1(C(CCC=C)=O)CCOC(CC(=O)N(C2CC2(C)C)C)C1 33130,C(CCP(C)(C)=O)NC(C1(N(C(=O)CCC2CCC(=O)C2)C)CC1)=O 33131,N1(C(c2n(CC)cnn2)=O)CC2CCCC2(NC(=O)Cc2n[nH]c(C)n2)C1 33132,C1(N(C(C)C(=O)OC(C)(C)C)C(C)=O)CCN(C(c2ncoc2C)=O)CC1 33133,C1(NC(C(C)NS(CC)(=O)=O)=O)CN(C(C2CCS2(=O)=O)=O)CCC1C(F)(F)F 33134,C(CC(C(=O)NC1CCN(C(C)=O)C1)NC(C1CCCSC1C)=O)=CC 33135,CC1(NC(C2CCCOC2)=O)CN(C(=O)C=Cc2ncco2)C1 33136,C1(F)(CNC(c2c(C)nco2)=O)CCCN(C(c2ccnn2C2CCC2)=O)C1 33137,CCC(C)C(CO)NC(=O)C(CC1CC1)NC(c1cc(C#N)cs1)=O 33138,CCC(C)CCCCC(=O)NOCC(=O)N(C(C(N)=O)C1CC1)C 33139,C(=O)(C(C)(C)CO)NC(C)C(C)NC(=O)CCOc1cccc(Br)c1 33140,C(=O)(CCCCC1CCCCC1)N(CCCN(C(CCCNC(=O)OC)=O)C)C 33141,C1(NC(CC(CC)C)=O)(CC)CCN(C(=O)CC23CCC(CC2)CC3)CC1 33142,Cc1cc(C(=O)Nc2ccccc2CN2CCC(n3cc(I)cn3)CC2)ccn1 33143,C1(N(C(c2csnn2)=O)Cc2nc(CC)sc2)CCN(CCCO)CC1 33144,CC1CC(NC(C2(CF)CCC2)=O)CN1C(=O)Cc1cc(C2CC2)on1 33145,c1(C(=O)NCC(CNC(=O)CCSC(F)(F)F)OC)cc(C(C)(F)F)ccn1 33146,N1(C(c2c(C)ncs2)=O)CCOC2(C1)CN(C(C1CC(C)(C)CO1)=O)C2 33147,n1(CC#C)c(C)cc(C(=O)NC2(CF)CCN(C(C3CC(F)C(=O)N3)=O)C2)c1C 33148,N1(C(c2n(C(C)C)ncc2)=O)CCOC2(C1)CN(C(=O)C(C)CS(C)=O)C2 33149,CCC(C(=O)OC)C(=O)NCC(CC)NC(=O)CC1(c2ccon2)CCC1 33150,c1(COC(C(=O)N(C2CCN(C(=O)CC3(OC)CCC3)C2)CC)C)ccncc1 33151,N1(C(C2(CC)CCOC2)=O)CCCC(C)(CNC(c2csc(CC(C)C)n2)=O)C1 33152,c1(OC)ccc(C(=O)NCCN(C)C(C2CN3CCN2CC3C)=O)c(OC)c1C 33153,C(=O)(CC1OCCc2ccccc21)N(CCCNC(c1csc2nnsc12)=O)C 33154,C1(OC)CC2CCC(C1)N2C(=O)CCCN(C)C(C1(C)CNC(=O)C1)=O 33155,c1(C(N(C2CCCN(C(C3C=CCC3)=O)C2)C)=O)cc(Br)cc2nc[nH]c12 33156,N1(C(COCCCOC)=O)CC2(C1)SCCC2NC(=O)C(O)P(C)(C)=O 33157,O=C(C1=CC2(CCOC2)C1)N1CCN(C(=O)C2=C(Cl)CCCC2)C(C2CC2)C1 33158,c1(C(=O)NCC2(NC(C(C)Cc3ccco3)=O)CCCC2)cn(C)nc1C1CC1 33159,c1(NC(C2CN(C(C3C=CCS3)=O)CC2C(F)F)=O)nccnc1-n1ccnc1 33160,CCC(C#N)(CC)C(=O)N1CC2CC1(CNC(=O)Cn1nc(C)ccc1=O)C2 33161,c1(C(=O)NCC(=C)CCNC(C23CCCCC2C3)=O)cc(C)cc(C)c1C 33162,N1(C(C(C)N(C(=O)CC(C)CC)CCC)=O)CC(CO)C(C)(C)C1 33163,C1(NC(C(Cn2cccn2)NC(C(C)N2CCCC2)=O)=O)CC2C(O)C(O)CC12 33164,c1(N(CCC2CCN(C(CCC3CCC(C)O3)=O)CC2)C)nccc(C#N)n1 33165,C(C)(CCC(=O)NC(c1nnc(O)n1C)C)NC(CCOCC)=O 33166,c1(C(N2CCC(NC(C(C)(C)CC#N)=O)(CO)C2)=O)cc(Br)cc(F)c1F 33167,N1(C(CCSC)=O)CCCC2(CCN(C(c3c(N)cc(Cl)cc3Cl)=O)C2)C1 33168,CN1N=CC(CC(N2CCOCC2CC(=O)NCCc2cccc(F)c2)=O)C1=O 33169,c1(C(N(CCN(C(=O)Cc2cc(Cl)cs2)C)C)=O)csc(S(N)(=O)=O)c1 33170,Cc1c(C(N2CCCC2Cn2cc(CC3(O)CCSC3)nn2)=O)sc2nccn12 33171,C1(C(N(CC(C(C)C)OC)C)=O)CC2(CC2)CN1C(c1cc(C)ccc1F)=O 33172,c1(C(N2C3CC(CNC(C(CCC)(C)C)=O)C2CC3)=O)cc2n(n1)C(C)CCC2 33173,c1(C(C(=O)NCC(C)NC(CCOc2ccc(C)cc2)=O)O)ccc(F)c(F)c1 33174,C(CC)(CCC(=O)N(c1cc(F)ccc1C)C)NC(CN(CC)CC)=O 33175,C(CC(=O)N1CCC(N(C)C(c2cc(C(C)(C)C)[nH]c2C)=O)C1)(C(F)(F)F)OC 33176,N1(C(C2C3CCC(F)C23)=O)CC2CCCC2(C(N2CCCCC2CO)=O)C1 33177,c1(C(=O)OC)nc(CNC(=O)CC(c2ccc(F)cc2)C)n(C)n1 33178,N1(C(CC(C=C)(C)O)=O)CC(NC(c2cnn(C(F)F)c2)=O)C(N=[N+]=[N-])C1 33179,C1(C)(CNC(CC2C=CC(NC(CC(C)SC)=O)C2)=O)CC(C)=NO1 33180,N1(C(C(C)SCC)=O)CCCC12CCCN(C(C1(C)CCCCCC1)=O)C2 33181,C1(N(C(CCc2onc(C)n2)=O)C)CCN(C(c2c[nH]cc2Br)=O)CC1C 33182,Cn1cc(C(=O)NCC(O)CN(C(=O)COCCCF)CCO)ccc1=O 33183,C(=O)(CC(C(F)(F)F)n1cccn1)NC(C(CC)C)CO.C12=CC=C(C=C1)C2=O 33184,c1(OCC(=O)NCC(CCOC)NC(C2CCOC(=O)N2)=O)c(Cl)cccc1Cl 33185,CCCC(C(=O)NC(C)CC)NC(=O)CC1CC2CC2C1 33186,C1(NC(c2cnc3[nH]nnc3c2)=O)CC2CN(C(c3occc3Cl)=O)CC2C1 33187,n1(C(C)C)ccc(S(=O)(=O)NNC(=O)c2ccc3c(c2)OC(F)(F)O3)n1 33188,c1(NC(C2C(NC(c3ccc(CNC(C)=O)cc3)=O)C2)=O)c(C=O)c(C)nn1C 33189,C1(C(N2CCC(CC)C2)=O)N(C(c2snnc2C)=O)CCC1(C)C 33190,c1(C(N(CCN(C(C2NC(=O)OC2C)=O)CC)CC)=O)ccc(C(C)C)cc1F 33191,c1(C(=O)NC(CCCC)CNC(=O)CCCCC(C)C)coc2cc(F)ccc12 33192,c1(OC)cc(C#N)ccc1-c1c[nH]nc1C(=O)Nc1ccc2c(c1)OCO2 33193,C1(C(=O)NC2CC(CNC(c3cn(C)c(=O)cn3)=O)C2)CCCC1S(C)(=O)=O 33194,CC1CCC(CNC(=O)CC2CN3CCC2CC3)CN1C(c1ccnn1C)=O 33195,C(CS(=O)(=O)CC(=O)NC1CN(C(=O)CCc2ccncn2)CC1(C)C)OC 33196,C1(NC(=O)CCc2ccco2)CC2CC1CN(C(c1noc3c1CCCC3)=O)C2 33197,C(=O)(C1c2c[nH]nc2CN1C(=O)C(CO)NC(=O)C1CC1)N(C(CC(C)C)CO)C 33198,C(CCNC(=O)CCc1cccnc1F)(C(C)(C)C)N(C(=O)CC(C)(C)C)C 33199,C1(N(C(c2c(C)nco2)=O)C)CCCC(NC(=O)C(c2cc(Br)co2)=O)C1 33200,N1(C(c2c(CC)nn[nH]2)=O)CCC2(CC1)CN(C(c1nnsc1C)=O)CC2CO 33201,N1(CC)CCN(C(c2cnn(C3CCOCC3)c2)C(=O)NC2CC2)CC1(C)C 33202,C12(C(N(CCN=c3[nH]ncs3)CC)=O)CCCCC1OCC2 33203,N1(C(C=CC(C)C)=O)CCC(NC(C2CCS(=O)(=O)C2)=O)C12CCC2 33204,CCCC(C(=O)NOC(CC(C)C)C(=O)NCc1ccc(F)cc1C)NC(N)=O 33205,C1(NC(C2C(C)C2C)=O)CC2CCC1CC2NC(C1CCC(=O)N(C)C1)=O 33206,c1(C(N2C(C3CCCN(C(C(=O)N(C)C)=O)C3)CCC2)=O)cccc(O)c1 33207,Cc1nc(NCC2(C)CCC(NC(C3CC3C)=O)CC2)c2c(C)csc2n1 33208,C1(C)(C(N(CC#C)CC=C)=O)CC(O)CN1C(c1cnnn1CC)=O 33209,C1(CN2CCC(c3n(Cc4sccc4)cnn3)CC2)COC2(CCC2)CO1 33210,C1(C2(O)CN(C(c3oc(SC)cc3C)=O)C2)(CNC(C(C=C=C)C)=O)CC1 33211,c1(OC)cc(CNC2CC2C(N2CC(OC)CC2CO)=O)c(Cl)cn1 33212,N1(C(Cc2ccc(C(=O)OC)s2)=O)CC(C)CN(C(=O)CNC(C)=O)CC1C 33213,c1(N2C(CCNC(c3n[nH]cc3Cl)=O)CCC2)cc(C(F)F)ncn1 33214,c1(C(N2CCN(C(=O)C=CBr)C(C3CCC3)C2)=O)cccc2nonc12 33215,C1(CNC(CSCC)=O)N(C(c2cc(C(C)(C)C)on2)=O)CCCC1(C)C 33216,C1(NC(=O)NCC=CCCC)CC(=O)N(c2ccc(OC)cc2)C1 33217,N1(C(C(CC)NC(C)=O)=O)CCCN(C(c2ncccc2C(=O)OC)=O)CC1C 33218,C1(NC(CCC(=O)N2CC(Cc3cn(C(C)(C)C)nn3)C2)=O)CC(C)(C)OC1=O 33219,C1(C(=O)NCC(CNC(CNC(=O)OCC)=O)F)CCCN1S(C)(=O)=O 33220,C1(C(=O)NC2CCC(OCC)CC2)C2CCC(C2)C1NC(=O)C1=CCCC1C 33221,N1(C(C=COCC)=O)CCC(NC(c2cc(Br)c(CC)s2)=O)CC1C 33222,c1(C(=O)NCC2CCN(C(c3c(C)nc(C)o3)=O)C2)c(C)cc(F)cc1Br 33223,N1(CC(=O)NCc2ccsc2)CCC(C2CNC2)CC1 33224,N1(C(c2n(CC)ncc2)=O)CC2CCCC1C2CNC(C1(C)CCCO1)=O 33225,C1(C(=O)NCC(CCC)(C)O)CCC2(CC2)N1C(C1CC2CCC2C1)=O 33226,Cc1ccc(NC(C2CN(C(c3sc(Cl)nc3Cl)=O)CCC2(F)F)=O)c(C#N)c1 33227,Cc1cc(CNC(C2(CCNC(=O)COCCCF)CC2)=O)c(C)s1 33228,C1(NC(CCC=CC)=O)CC(O)CN(C(c2cnn(C3CCCCC3)c2)=O)C1 33229,C(=O)(C(O)C(C)(C)C)NC1CC(CC(=O)NCCNC(N(C)C)=O)C1 33230,C1(C(=O)OCC)C2C=CC(CC2)C1C(N1CC(C)(C(=O)OC)C1)=O 33231,Cc1ccc(C(C)C(=O)NCC2CN(C(=O)C=Cc3cn(C)cn3)CCO2)cc1 33232,n1(CCC)cc(C(=O)NCc2c[nH]nc2C2CCN(C(=O)C(F)OC)C2)cn1 33233,Cc1cnc(C(=O)NCC2CCCN(C(c3cncnc3C)=O)C2)cc1C 33234,C1(CNC(C(C)N(CC)CC)=O)(CO)CCCN(C(c2nc(C3CC3)cs2)=O)C1 33235,Cn1ccnc1SCC(=O)NCCCN(C(C1(O)COC1)=O)C1CC1 33236,c1(C(N2CCC(C)(NC(C(C)n3ccnc3)=O)CC2)=O)ccc2sncc2c1 33237,N1(C(CS(C)(=O)=O)=O)CCC2CCC12CNC(=O)CCOc1ccc(F)c(Cl)c1 33238,CCC(F)(F)CC(=O)NCCn1cc(C(=O)NCC2CC(=O)NC(C)C2)nn1 33239,N1(C(C2N(C(=O)CN3CCC(C)C3)CCC(C)C2)=O)CCCC(C2(C)CC2)C1 33240,N1(C(CCNC(=O)NC)=O)C2CCC1CC(NC(=O)CC1(CSC)CC1)C2 33241,C12CC(C(O)C1)N(CC)C2=O.c1(CN2C(C(=O)NC)CCC2)cccnc1 33242,Cn1cnc2cc(CC(=O)NCC3CC(NC(C4CCCC4)=O)C(O)C3)ccc12 33243,C(C(=O)N(CC(C)(C)CNC(c1nocc1C1CC1)=O)C)(C(C)C)SCC 33244,C1(C(N(C)CC)=O)(COC)C=CCN1C(c1cn(CCN2CCCC2)nn1)=O 33245,CN1N=C(C(=O)NCC2CCCN(C(=O)C(C)(C)CCF)CC2)CCC1=O 33246,C1(CC(=O)N(CCN2CCN(C(C3(CCC)CC3)=O)CC2)C)CCCC(C)(C)O1 33247,C1(C)(C(N2CC(SC)C(NC(C3(C(=O)N(C)C)CC3)=O)C2)=O)CC2(CCC2)C1 33248,c1(C(=O)NCCC(=C)CNC(=O)C(C)(C)C(=C)Cl)cc2nc(C)cc(C)n2n1 33249,C1(C(N2CCC(N(C(=O)C(C)(C)C3CCCCO3)C)C2)=O)C(C)(C)OC1(C)C 33250,N(C1CCc2c(F)cc(F)cc21)C(c1c(OC)c(Cl)cc(C)c1)c1nnnn1C 33251,N1(C(c2c(C)ccnn2)=O)CC(F)(F)CC1CNC(=O)C(N1C(=O)CCC1=O)C 33252,n1(CC#C)cnnc1C(=O)NC(C1CCOC1)CNC(=O)CNS(=O)(=O)CCC 33253,c1(CC)nc(C)c(CC(=O)NC(C)(C)CNC(=O)C=CSc2nc[nH]n2)c(C)n1 33254,c1(C(=O)NC(CNC(c2cc(C)ncc2)=O)(C)C)cc(N2CCCC2)nc(Cl)c1 33255,CCS(=O)(=O)CC(=O)N1CC(CNC(c2cc(F)n(C)n2)=O)CC1C 33256,N1(C(C=C(CCN(C)C)Cl)=O)CCOC2(C1)CN(C(C1CCCN1N=O)=O)C2 33257,c1(C(=O)NCC(=C2CN(C(C3CC3(F)F)=O)C2)F)n[nH]c(C2CC2)n1 33258,C1(C(N2CCC(CNC(C(C)(C)Cc3cnn[nH]3)=O)CC2)=O)CN2CCN1CC2 33259,N1(C(c2c(CC)csc2)=O)Cc2ccccc2C(NC(C2CCNC2=O)=O)C1 33260,C(=O)(C1CSc2ccccc21)Nc1ccc(C(=O)OC)c(OC(F)(F)F)c1 33261,N1(C(c2c(CC)noc2C)=O)CC(CC(=O)NCC(C)(O)CC)C2(CC2)C1 33262,c1(NC(=O)C2CC2)ccc(CNC2CCCC2Oc2ccccc2)cn1 33263,C1(C(=O)NCC2(C(N)=O)CN(C(c3ccc(F)c(Cl)c3)=O)C2)CC2C(C1)C2(C)C 33264,C1(C(=O)NCCC2(CO)CC2)(Cn2cc(COCCO)nn2)CCCCC1 33265,C1(NC(c2c(CC)ocn2)=O)CCCN(C(=O)C=CC2CC2)CC1F 33266,c1(CC)cnc(O)c(C(=O)N(C)CC2CCCN2C(c2n[nH]cc2OC)=O)c1 33267,N1(C(C2CC3CC3C2)=O)CCC2(C1)c1[nH]cnc1CCN2C(C1(O)COC1)=O 33268,CC(C)CC(CNC(c1cocc1C(N)=O)=O)C(=O)NC(C)CC1CCC1 33269,c1(OCCC)cccc(C(=O)NC2CN(C(=O)C(C)=C3CCC3)CC2C)c1 33270,CCCC(CCCNC(=O)CC1CCCCCO1)NC(=O)CNC(=O)C(C)(C)C 33271,N1(C(c2scc(CNC(c3c(C)ocn3)=O)c2)=O)C2CCC1COC2 33272,Cc1cc(C(=O)N(C2CCN(C(c3cnc(N(C)C)o3)=O)CC2)C)c(C)nc1C 33273,c1(C(=O)NCC2CC(NC(CC3CCCC(C)(C)O3)=O)C2)cccc2nncn12 33274,C1(F)(CNC(CCOCCOC)=O)CCN(C(c2cnc(S)nc2)=O)C1 33275,N1(C(C2C3(CN(C(c4c(C)nn(C)c4C)=O)C3)C2)=O)C2CCC1CN(C)C2 33276,c1(CC(=O)OC)cccc(Br)c1NC(=O)C(=O)NCc1ccn(C2CCCC2)n1 33277,CC1(C)Cn2[nH]c(=NC(=O)NCC3CC(F)(F)C(=O)N3)cc2CO1 33278,CN1CCC(NC(C2CCC(NC(C3(N(C)C)CCC3)=O)C2)=O)C(C)(C)C1 33279,c1(C(c2n(C)nnn2)NCC(C)(C)OCCO)cc(Br)c(Br)o1 33280,C(=O)(CC(C)(C)C)NC(C)C(N1CCC(N(c2cc(Cl)ncn2)CCO)CC1)=O 33281,N1(CC)CCOCC1C(=O)N(CC(O)CN(C(=O)CCN1CCNC(=O)C1)C)C 33282,C(CCN=C(NCc1cccnc1Cl)NC1CSC(C(F)(F)F)C1)SC 33283,c1(CC)cccc(C(=O)OC)c1NC(=O)CN1CCOCC1C1CCCOC1 33284,c1(C(N(C(CC)CNC(=O)C(F)OC(F)(F)F)C)=O)cccc2nsnc12 33285,C(CCC(=O)NCC(CC)NC(=O)C(C)CNC(=O)OC(C)(C)C)=C(C)C 33286,C1(C(=O)NC2(CNC(c3cnsc3)=O)CC2)CCc2nnc(O)n2C1 33287,c1(CN(C(=O)CC(C)(C)C2CC2)C)cc2sccc2[nH]1.C12CCC(CC1)CN2 33288,N1(C(C2C(NC(C3CC4(CCC4)CO3)=O)CC2)=O)CCC2(CC1)CC2CO 33289,C1(CNC(c2c(C)nc(O)[nH]2)=O)CN(C(=O)CC2CCC3(CCC3)O2)CCN1C 33290,N1(C(c2c(C)cn(C)c2)=O)CC(C)CN(C(=O)Cn2cnc(Br)c2)CC1C 33291,C(=O)(C(C)(O)CC)N1CC(CCO)(CNC(CCCOCCOCCCC)=O)C1 33292,C1(NC(C2C(CCC)C2)=O)CN(C(c2ccc(-n3cnnn3)cc2)=O)C(C)(C)C1 33293,C(CCS(C)=O)(C(=O)N1CC2C(NC(c3ccc(O)cn3)=O)C2C1)N(C)C 33294,c1(CC)onc(C(=O)NCC2(C)CCN(C(c3ncc[nH]c3=O)=O)C2)c1C 33295,C1(C(=O)NCCn2ccc(C(=O)NCC=CCCOC)c2)C2CCC(C2)C1C 33296,C(=O)(C1CCCc2ccnn21)N1C(C)CC(NC(C2(OC)CCS(=O)(=O)C2)=O)C1 33297,Cc1nccnc1C(=O)NC1(CC=CC(=O)NCC2(OC(C)C)CCC2)CCC1 33298,c1(C(=O)NCCCN(C(=O)CP(C)(C)=O)CC)c(C)nc2ccccn12 33299,c1(C(=O)NC2C(C)CN2C(=O)C=Cc2ccco2)ccnc(OCCO)c1 33300,C(CC1=CCOCC1)NC1(c2nnnn2CSc2ccccc2)CC(CCF)C1 33301,N1(C(CNC(c2cc(C(C)(C)C)[nH]c2C)=O)=O)CCCCC1C.CC(=O)OC 33302,C1(CNC(CCc2cnc(C)s2)=O)CN(C)CCN1C(=O)CCc1cnc[nH]1 33303,N1(C(C(CC=C)(C)O)=O)CC=C(C(=O)N(C)Cc2nc[nH]n2)CC1 33304,CC(=Cn1ccnn1)C(=O)NCC12CCC(CN(C(c3cccnc3O)=O)C1)C2 33305,N1(C(Cc2cc(C)on2)=O)CC2(CCN(C(=O)CCC3CCCC(O)C3)CC2)C1 33306,c1(OC)cncnc1C(=O)N(C(C)C(=O)NC1CCCCC1F)C1CC1 33307,C1(C(=O)OC)CCN(CC(=O)N(C)CC2CC2)CC1.N12CCCC1C2 33308,c1(C(=O)NCC(CNC(C2N(C(C)=O)CCC2)=O)O)cc2c(O)ccc(F)c2[nH]1 33309,c1(C(N(C(CNC(c2c(OC)n[nH]c2)=O)C)C)=O)cc2c(nn1)CCCC2 33310,C(=O)(C(C(C)(C)C)NC(c1ccnc(CNC(c2cnc(Br)s2)=O)c1)=O)NC 33311,CCN=c1[nH]cc(C(=O)NC2COCC2NC(c2nc(C)oc2C)=O)s1 33312,c1(CN2CC3N(C(C4CCCN(C)C4)=O)C(C3)C2)c[nH]c2ncc(Br)cc12 33313,N1(C(C2C(C)(C(F)F)C2)=O)C(C(N2CC(N3CCCCC3)C2)=O)CCC12CC2 33314,C1(NC(C2C(=C)CC2)=O)CCSC12CN(C(c1cnn(C3CCC3)n1)=O)C2 33315,CC1(C(=O)NCC2CCCCN2C(c2ccn(C3CCC3)n2)=O)CC2CCC1C2 33316,CCC(CC(F)(F)F)C(=O)NC(CC)(CC)CCNC(=O)CNC(=O)CC(C)(C)C 33317,N1(c2n(CC=C)c(C(O)CCOC)nn2)CCC(C)CC(C)C1 33318,C1(NC(c2c(C)con2)=O)CN(C(=O)Cc2ccns2)CCC12CCC2 33319,Cc1cc(C(N2CCN(C(c3ccccc3OC(F)F)=O)CC2)=O)nc(CO)n1 33320,Cc1nc2sn(CCC3CCS(=O)(=O)CC3)c(=O)c2c(C)c1C 33321,C1(NC(c2cnc(C)o2)=O)CCOC12CCN(C(c1cc(Br)c[nH]1)=O)CC2 33322,N1(C(c2nc(CCC)sc2)=O)CC2ON=C(CNC(c3nc(C)oc3C)=O)C2C1 33323,CC(C)CC(CNC(C1(F)CC1)=O)NC(C1(CC2CC2)CC1)=O 33324,CCCC(C)(O)CC(=O)N1C2CCC1C(CNC(=O)CC1(C(F)(F)F)CC1)C2 33325,N1(C(=O)CCc2nccs2)CCCCC1C(N1CCOC2CC12)=O 33326,c1(CC(=O)NC(C(C)NC(c2cc(C)c(C)nn2)=O)C)ccc2ncsc2c1 33327,c1(C(C(=O)N(C)CC2N(C(CN(C)CC)=O)CCC2)O)cccc(C)c1 33328,N1(C(C(C(=O)OC)(C)C)=O)CC2CCN(C(c3nc(C4CC4)cs3)=O)CC2C1 33329,N1(C(CC(=O)NC2CC2)=O)CCC(C(=O)NCc2cccc(F)c2)C12CCC2 33330,N1(C(CC(CC)OC)=O)CCCCC2(CCN(C(=O)OC(C)(C)C)C2)C1 33331,c1(NC(CN2CCCC(C(C)NC(C(C)C)=O)C2)=O)ccc(F)c(Br)c1 33332,c1(C(CC)(C)NC(=O)C=CCN(C)C(C2(n3cncn3)CC2)=O)ccc(F)cc1 33333,Cc1cc(CN2CC(F)(F)CC2C(=O)Nc2nc(Cl)nc(Cl)n2)cnc1Cl 33334,C=CC(CCC)CC(=O)NC12CCC(NC(=O)C(O)CC(F)(F)F)(CC1)C2 33335,N1(C(CC2(C(=C)F)CCC2)=O)CCC2(CNC(=O)CCC3CCC3)CCCCC12 33336,N1(C(CC(C)(C)n2cc(C3CC(=O)C3)nn2)=O)CC(CC(=O)O)OCC12CC2 33337,C(C)(C)(CCCNC(=O)C(C)(C)C1CCCN1C(=O)CC(C)SC)OC 33338,CCCCCC(O)CC(=O)N(CCCCN(C)C(c1ccccc1N)=O)C 33339,C1(OC)CC(CC(=O)NCCC2CN(C(=O)CC(C)C)CCO2)C1(C)C 33340,N1(C(c2scc(C)c2)=O)CCC2(CC1)OCCC2NC(=O)C(F)C1CCC1 33341,C(=O)(CCC1=NNC(=O)CC1)NCCC(=O)NC1(C)CC(NC(=O)CO)C1 33342,S(=O)(=O)(c1cc(F)cc(Br)c1)N(C(=O)C(C)Oc1ccc(F)cc1)C(C)C 33343,N1(C(C(CSC)O)=O)CCC=CC1C(=O)N(CCO)CC1CC1 33344,c1(N2CCCC3(NC(c4ncc(F)cc4F)=O)C(C2)C3)ncc2cccnc2n1 33345,C(C)(C)(CCCCNC(C1(n2nccn2)CC1)=O)NC(C(CSC)OC)=O 33346,c1(C(N2CC=CC(NC(c3c(C)ccc(C)c3)=O)C2)=O)nn(C)c2c1CCCC2 33347,c1(C(=O)NC(C(C)(C)NC(Cc2cc(C(C)C)no2)=O)C)cncnc1C1CC1 33348,c1(C(=O)NCCC(CNC(c2n(C)nc(C3CC3)c2)=O)O)ccc(F)cc1O 33349,C1(C(N2CCC(C)(C)C2)=O)CCCN(c2ccc(Br)cc2)C1=O 33350,N1(C(CCC=C)=O)CCc2ccccc2C1CCNC(c1cnc(Cl)s1)=O 33351,N1(C(C(COC)C)=O)CC(NC(c2cc(=O)n(C)o2)=O)CC12CCCCC2 33352,C1(C2CC2)(CNC(C(C(C)O)NC(C)=O)=O)CCN(C(=O)C2=C(C)OCC2)C1 33353,C=CC1CC(NC(c2ccccc2-n2cc(COC(=N)O)nn2)=O)CCO1 33354,c1(CSC)cccnc1C(=O)N(CC(C)N(C(=O)Cc1cnc(C)[nH]1)C)C 33355,CCC(O)C(C)C(=O)NC1CCC(CNC(c2cccc(C#N)c2)=O)CC1 33356,N1(C(c2c(SC)csc2)=O)CCCC(NC(=O)CC2CC2(C)C)C1 33357,C(=O)(CS(=O)(=O)C1CC1)NC(C(C)C)CCN(C(=O)Cc1ccn(C(F)F)n1)C 33358,Cc1cncc(NC(c2cnc(CNC(=O)CC3CSCCO3)nc2)=O)c1 33359,CCC(C)(C(=O)N1CC(O)(CCNC(=O)Cc2ncc(F)cc2F)C1)C(N)=O 33360,CN1CC(C(=O)NCC(C)(C)NC(=O)C=CC(N)=O)CCC1=O 33361,N1(C(C(C(C)C)NC=O)=O)CCC2(CCN(C(c3ccc(O)c(N)c3)=O)C2)C1 33362,c1(-c2n(CC3CN(CC(F)(F)F)C3)nc(C3CCC3)n2)nc2ncc(Br)cn2n1 33363,C1(C(N2CC3CCC(C2)N3C(=O)CCSC(F)(F)F)=O)CCCC2CCCN12 33364,C1(CNC(C2N(CC)CC2)=O)CCC2(CCC2)CN1C(=O)C(Cl)=CCl 33365,c1(CC)nnsc1C(N1CC(CC(C)NC(c2cnn(CC(F)(F)F)c2)=O)C1)=O 33366,c1(OCC(NOCCCC(=O)OC)=O)cccc(C#N)c1 33367,C1(CCNC(c2cscn2)=O)CCN(C(c2cc(O)ncc2F)=O)CCC1(F)F 33368,c1(C(N2C3CC(OC)(C3)C2)=O)cccc2ccn(C)c12 33369,Cc1cc(Cl)nc(N)c1C(=O)NCC1CC(C)CCN1C(C1CCCN1C=O)=O 33370,C(=O)(CCCCCNC(C1CC12CCCCC2)=O)N1CCN(CC#CC)CC1 33371,Cc1ccc(CNC(C2C3CN(C(=O)CCc4ccoc4)CC23)=O)c(O)n1 33372,c1(C(=O)NCCCC(C)NC(=O)C2CC2)cccc(OCc2ccccc2F)c1 33373,CCCC(C#N)NC(C12CC(n3cc(C4CCC4)nn3)C1C2)=O 33374,C1(C(N(CCCNC(c2ccnn2C(C)C)=O)CC)=O)CCCC(CF)C1 33375,C(c1ccoc1)=CC(N1CCC(NC(=O)C(F)(F)F)C1)=O 33376,C1(C(C)C)CC(CC(=O)N(C)CCN(C)C(C2CC(=C(F)F)C2)=O)CCO1 33377,N1(C(Cc2cc(C)ns2)=O)CCCN(C(=O)CCC(CF)CF)C(C)C1 33378,c1(N2CC(C)C(CO)CC2)nccc(=NCCc2cccc(N)c2)[nH]1 33379,N1(C(CN(CCCCCC)C)=O)CC(NC(=O)C=CC(C)(C)C)C2(CCC2)C1 33380,c1(NCC2(NC(CCOCC#C)=O)CCC2)nccc(Oc2ccccc2F)n1 33381,c1(C(N2CC(NC(c3c(C)n(C)nc3)=O)C(C)C2)=O)cnc2sccc2c1 33382,C(C(CC(F)(F)F)NC(c1cccc(O)c1Cl)=O)NC(C(CC)N(CC)CC)=O 33383,N1(CCC)C(=O)CCC1C(N1CCCCC1CCNC(c1ncncc1Cl)=O)=O 33384,C#CCCC(O)C(=O)NCCCN(C(C1(C(=O)NC)CC12CC2)=O)C1CC1 33385,C1(C(N2CCC(C)(NC(c3cc(C)c(C)o3)=O)C2)=O)CCCC2(CCC2)O1 33386,N1(C(c2ncccc2C)C(=O)NC)CC2CC3CC2C1C3O 33387,C1(CNC(c2cnnn2C2CC2)=O)CN(C(C2C3(CC3)C23CC3)=O)CC12CC2 33388,CC1CC(C(=O)N2CC(O)(C3CCCN3C(=O)C#CC3CCC3)C2)=NO1 33389,CC1CN(C(=O)C(c2ccc(Cl)cc2)O)CC1NC(=O)C(C)C1CCOC1 33390,C1(CNC(=O)CC2CCOC2)C=CCN1C(=O)CCCN1CCCCC1 33391,c1(CCCCN(C)C)ccccc1.C1(=O)C=CC(=O)NC2C(C2)C(C)N1 33392,c1(CC)ccc(C(=O)NCC(CCOC)NC(=O)CC=C(C)C)o1 33393,C1(NC(c2c(CC)noc2C)=O)CC2CC(NC(=O)C(C3CCOCC3)F)C2C1 33394,Cc1cccc(C(=O)NCC2CC(C(=O)N3CC(C)(C#N)C3)=NO2)c1C 33395,Cc1ccc(CNC(C2C(O)CCN2C(C2CCC(C)(C)OC2)=O)=O)c(O)n1 33396,N1(C(C(C#N)C2CC2)=O)CCOC2CN(C(c3c(F)cccc3F)=O)CC12 33397,C#CCCCCCC(=O)NC(C)(CNC(C1CC1c1ccccc1Cl)=O)C(C)C 33398,c1(C(N2C3(CNC(CC4C(C)CCCC4)=O)CC(C2)C3)=O)cc(F)ccc1N 33399,C(=O)(CC(C(F)F)NC(c1conc1C)=O)N1CCC(O)(CC)C1 33400,N1(C(c2cncc(OC)n2)=O)CC(C(=O)NCC(O)C(C)(C)C)CC(C)C1 33401,N1(C(C(C)=C2CC2)=O)CC(N(C(=O)Cc2c[nH]nc2C)C)C(C)(C)C1 33402,N1(C(c2cc(C)[nH]c2C)=O)C2CCC1CN(C(c1cccc(C3CC3)n1)=O)C2 33403,CC1=C(C)CC(C(=O)NCC2COCCN2C(c2csc(C)c2C2CC2)=O)CC1 33404,N1(C(C(C2CCOC2)NC(c2nc(CCC)oc2)=O)=O)CCC12CCCC2 33405,c1(C(=O)NC2CC(NC(c3coc(Br)n3)=O)C2)ccc(-n2ccnc2)cc1 33406,c1(COCC)nc(C(=O)NC(C)(CNC(c2ccc(Cl)o2)=O)C2CCC2)cs1 33407,c1(CN(CC(C)CS(C)(=O)=O)C)c[nH]c2cccc(Br)c12 33408,Cc1ncnc(C(N2CCC(C)(NC(c3cccc(Br)c3)=O)C2)=O)c1C 33409,C(C(C)C(C)C(=O)NCC(C(C)(C)C)NC(=O)COC(F)F)OC 33410,C1(C(=O)NCCn2c(C)cnn2)CCC(C)(C)N(C(=O)COCCCN(C)C)C1 33411,C1(O)(CCNC(C=CC(C)(C)SC)=O)CCN(C(=O)CC2C=CCCC2)C1 33412,c1(C(N2C3C(NC(c4c(Cl)ccc(SC)c4)=O)C(C3)C2)=O)c(N)ccc(F)c1C 33413,C1(C(=O)NC(CC)(CNC(c2n[nH]c(C)c2Br)=O)CC)CCC2CC2CC1 33414,C12(NC(CNC(C)=O)=O)CN(C(C3(Br)CC3)=O)CC1CS(=O)(=O)C2 33415,C1(NC(c2c(OC)noc2C)=O)CC2CC1CN(C(c1ccccn1)=O)C2 33416,C1(NC(CN(C2CCSC2)C)=O)CC2CC(C1)N(C(=O)CC1CCCC1(F)F)C2 33417,C(=O)(C1=CCOCC1)NC1CC(C(C)NC(C2CC(=C3CCC3)C2)=O)C1 33418,C1(CN(C(C2CC(N3CCC3)C2)=O)CC)CCCN(C(c2cscc2C)=O)C1 33419,C1(CC(=O)NCC2(CNC(c3ncc(C)cn3)=O)CCCC2)(OC)CCOCC1 33420,C(=O)(CCCC(C)NC(=O)COC(C)(C)C)NCC(COC)(C)O 33421,Cc1ccc(C=CC(N2CC(C3(NC(c4ccc(F)s4)=O)CC3)C2)=O)cn1 33422,N1(C(CC)=O)CCC2(CC1)CC(NS(=O)(=O)CCOC)C2 33423,Cc1cn2cc(C(=O)NCC3CC(F)(F)CN3C(=O)C(C)N(C)C)cc(F)c2n1 33424,c1(C(=O)NCC(C)NC(c2c(OC)ncc(Br)c2)=O)cnc2ccnn2c1 33425,C(=O)(CC(O)CC(C)(C)C)N1C2CCC(NC(c3nc(OC)c(F)cn3)=O)(C2)C1 33426,C1(CC#C)(C(=O)N(CCNC(=O)CCc2cnoc2)C2CC2)CCCOC1 33427,C1(CC=C)(NC(C2CC(N(C)C)C2)=O)CN(C(c2cc(C3CC3)on2)=O)C1 33428,C1(CC#C)(C(=O)NC2CC2)CCCC1.C(C(C)O)CC 33429,Cc1cc(C(N2CCCCC2CNC(C2(n3cccn3)CC2)=O)=O)ncn1 33430,C1(C(=O)NC(CNC(c2cccc(SCC)c2)=O)CO)NC(=O)OC1(C)C 33431,CCC(C)C(C(=O)NC(CCO)CC(C)C)NC(=O)Cc1c(C)cnn1C 33432,N1(C(C(CC)NC(N)=O)=O)CCN(C(=O)CC2(C#N)CC2)C(C2CCCCC2)C1 33433,C(N=c1cc(C(C)(C)C)nc[nH]1)C1CN(C(c2cccc(C)n2)=O)CC1(C)C 33434,c1(C(C)C)ncc(C(c2nnnn2CC(F)F)NCC2CCCCC2)[nH]1 33435,N1(C(C(OC)OC)=O)CCCC(O)(CCNC(C23CC2COC3(C)C)=O)C1 33436,c1(C(N(CC(CC)NC(=O)CCC=C(C)C)CC)=O)cc(Br)c(OC)s1 33437,N1(C(C(C)(C)OC)=O)CCC(C(=O)Nc2cccc(F)n2)C(c2ccccc2)C1 33438,c1(NC(=O)NCC23CC(C(F)F)(CO2)C3)nccc2cc(Br)ccc12 33439,CC1=C(C(=O)NC(C)CC2CCN(C(C3(C)CCCO3)=O)CC2)C(C)(C)CCC1 33440,c1(C(c2cn(CC(c3ccccn3)N(C)C)nn2)O)ccc(Cl)cc1 33441,C(=O)(CC(C)C(F)F)NCC(C)NC(=O)Cc1cccc(OC(F)F)c1 33442,Cc1ccc2c(C(=O)NCCCNC(=O)C(C(C)C)c3cnn(C)c3)n[nH]c2c1 33443,c1(CN)ccc(I)c(O)c1.Cc1cc(CNC(=O)NCCN)on1 33444,CN1CCN(C(=O)C(F)C2CCCC2)CC1C(=O)NCC1CC12CC2(F)F 33445,C(C1CCCc2cccnc21)NCc1ccc(Cn2cncn2)cc1 33446,c1(OCCC(=O)N(CCn2c(C)ncc2)C2CC2)cc(F)ccc1F 33447,c1(N(C(C(n2c(C)nnn2)c2ccccc2)=O)C)cc(F)cc(Cl)c1 33448,N1(C(C(C)(C2CCC2)NC(C(C)NC=O)=O)=O)CCn2ccnc2C1 33449,c1(CC2(N(C(C=CCC)=O)C3CC3)CCC2)nc(C(=O)NC2CCC2CO)co1 33450,n1(CC(=O)NCC2COCC2NC(=O)C(O)CC(F)F)cc([N+](=O)[O-])ccc1=O 33451,C1(C(=O)NC(C)CC(C)NC(c2sccc2F)=O)(Cc2cnn[nH]2)CCOCC1 33452,C12(NC(CCN(C3CCCCC3)C)=O)CC(C1)N(C(c1ccncc1Br)=O)C2 33453,c1(C(CC(=O)O)NCc2cccc(C3CC3)c2)cccc(F)c1Br 33454,C1(COC)(NC(=O)C(C2CC2)SC)CCCN(C(C2(O)COC2)=O)C1 33455,CC(C)C#CC(=O)NC12CC1CN(C(C1CCCN1C1CCOCC1)=O)C2 33456,c1(NC(CN(CC(C)C)C(=O)Cn2cnnn2)=O)ccccc1CCO 33457,N1(C(C(C)=C(CC)C)=O)CCCC2C1CCN2C(=O)C(C(C)(C)C)NC(N)=O 33458,N#Cc1cnc(C(F)(F)F)cc1NC1CCC(OCCO)CC1 33459,C#CCCCC(C)C(=O)NC1CC(C)N(C(c2ccc3nccn3c2)=O)C1 33460,C1(N(C(C(C)NC(CC)CC)=O)CCOC)CCOCC1 33461,CCC(CN(C(=O)C(C)OCOC)C)NC(=O)C=CC(=O)OC(C)(C)C 33462,c1(C(=O)OCC)cc(COC(C23CCC(C(F)F)(CC2)CC3)=O)ccc1[N+](=O)[O-] 33463,c1(CC(=O)NCCC2(NC(=O)CCc3cc(Cl)no3)CCCC2)cccnc1 33464,c1(C(=O)NCC(CC)NC(=O)C(C)OCCC(C)C)ccnn1CCOC 33465,c1(OC)cc(F)c(C(=O)NC2COCC2NC(=O)CC2CC=CC2)c(F)c1 33466,N1(C(C=C(COC)C)=O)CC2CN(C(=O)CC3CCCC34CC4)CCC12 33467,CC1CCCCN1CC(=O)N(C(=O)COc1ccc(C(N)=O)cc1)C1CC1 33468,c1(C(=O)O)ccnc(-n2ccnn2)c1.C1COCC1NC(C1(C(C)C)CCC1)=O 33469,c1(C(C)C)nn(C)c(NC(=O)CC2CCCC(NC(c3cccnc3)=O)C2)c1Cl 33470,c1(OC)cc(Cl)c(Cl)cc1C(=O)NCCC(C)NC(C1C=CCC1)=O 33471,C1(NC(COC(CC)(C)C)=O)CCC2(CC2)N1C(=O)CN(C(=O)COC)C 33472,C1(C)(N(C)C)CCN(C(C2CC(=O)CN2C(C2CCCN2C2CC2)=O)=O)C1 33473,C1(C(N2C(CNC(=O)C#CC(C)C)CC(OC)C2)=O)Cc2ccc(C)cc2S1 33474,c1(C(=O)NCCCC(C)(C)NC(c2c[nH]c(=NC)o2)=O)c[nH]c2c(Cl)cccc12 33475,C=C(Cl)C(C)(C)C(=O)NCC(O)CCNC(C1CC1CCC)=O 33476,C1(CNC(CCSCCC)=O)CC2(CO1)CN(C(=O)CCC=C(C)C)C2 33477,c1(CC)c[nH]cc1C(=O)NC(Cn1cncn1)C(=O)NCCCF 33478,CC1SCCCC1C(=O)NCCN(CCCN(C)C)C(=O)CC1(C)CC1 33479,C(=O)(C(C)(C)NC(C)=O)N1CC(C(C(=O)NCCCN(C)C)OC)C1 33480,CC1=NS(=O)(=O)NC=C1C(=O)N1CC(CCNC(C2CCCC3CCCN23)=O)C1 33481,c1(C(N2C(C(=O)NCC3(O)CC(C)(C)C3)CC(O)C2)=O)cc([N+](=O)[O-])c[nH]1 33482,C12(C(N3CC(CNC(c4c(C)csc4)=O)OCC3)=O)CC1CCC2(F)F 33483,Nc1ccc(F)cc1C(N1CC2CC2(CNC(=O)CCC2CCCCCC2)C1)=O 33484,C1(NC(c2cc(F)c(F)c(F)c2)=O)CC1C1CCCN(C(c2coc(O)n2)=O)C1 33485,C1(NC(=O)CCc2cc(F)ccc2Br)CN(C(C2(F)CC2)=O)CC(F)(F)C1 33486,N1(C(C(C(C)C)n2cnnc2)=O)CCN(C(=O)C(N)=O)CC(O)C1 33487,CC1CN(C(=O)CCc2cn[nH]c2)CCC1NC(=O)CCc1cnn(C)c1 33488,c1(C(N2CC(C(=O)Nc3cc(Cl)ncc3Cl)C2)=O)ccc2c(c1)CCO2 33489,c1(C(N2CC(N(C)C(c3cc(F)cnc3O)=O)C(F)C2)=O)c(F)ccc(F)c1Cl 33490,c1(C(N(C(C)CCNC(=O)C=CC2C(C)C2(Cl)Cl)C)=O)n[nH]c2c1CCCC2 33491,c1(CC)nnc(C)cc1C(=O)NCC1CN(C(c2cnc3n2CCC3)=O)CCO1 33492,C(=O)(C1COc2ccc(Cl)cc21)NC1C(CNC(c2c(CC)occ2)=O)CCC1 33493,N1(C(C2CCC(CNC(C3CC4CCC3O4)=O)CC2)=O)CCC(O)C(F)C1 33494,C1(C(=O)NCCC2CCCN2C)(NC(C(C=C)O)=O)CCCCC1 33495,N1(C(C2C(C)=C2)=O)CCc2ccccc2C(NC(c2cc(C(F)(F)F)on2)=O)C1 33496,c1(C(=O)NCC(c2ccc(Cl)cc2)NC(C(C)O)=O)cnc(O)cc1C(F)(F)F 33497,C(=O)(C1c2c[nH]nc2CN1C(C1CCC(F)CC1)=O)NCc1c(C)cc(C)nc1 33498,C1(CC(=O)N(CCCCCNC(c2c(C)cncc2)=O)C)CC2CCC1CC2 33499,c1(N(C)Cc2c(C)ccc(Cl)c2)nc2c(c(=NCCC3CC3)[nH]1)SCC2 33500,CCC(C)C(O)C(C)C(=O)NCC12CC(CO1)N(C(C1(C)CCC(=O)C1)=O)C2 33501,N1(C(Cc2ccn(C)n2)=O)CCCC(C)(C)C1CNC(=O)Cc1ccsn1 33502,CC(C)(C)CCC(=O)NCCCC1CCCCN1C(C1CCC2(CCC2)C1)=O 33503,c1(NC(c2cnc(OCC)c(-c3ccsc3C#N)c2)=O)c(Cl)cccc1[N+](=O)[O-] 33504,Cn1ccnc1N(CCO)Cc1cc(Nc2ccccc2)cs1.C12CCN(C1)C2 33505,C1(CNC(CCc2ncc(C)[nH]2)=O)CC(NC(c2sc(C)cc2Cl)=O)C1(C)C 33506,n1(C(C(=O)OC)C)cc(CN(C(CCCNC2CCC2)=O)C)nn1 33507,C1(C(=O)NCC(CNC(c2cn(C(C)C)nn2)=O)C)CCCC(=O)O1 33508,C1(NC(C(C(C)C)SCC)=O)CC2(CCN(C(=O)C=CCOC)C2)C1 33509,Cc1nc(C(=O)NCCCN(C(C2CCC(=O)NC2)=O)C2CC2)c(C)s1 33510,C1(NC(CONC(C(C)N(CC)CC)=O)=O)C2CCCC1COC2 33511,C(=O)(C(O)CCS(C)=O)N(C(C)C)CCNC(c1sccc1OC(F)F)=O 33512,C1(C(C)C)C(NC(=O)Cc2cncs2)CCN1C(C1OCCO1)=O 33513,Cc1nn(CC(=O)NC2CC2NC(C2(C)CC(C)(C)C2)=O)c(C)c1Cl 33514,c1(C(=O)NC2(CNC(CP(C)(C)=O)=O)CC2)cc2cc(Cl)cnc2[nH]1 33515,c1(CC(=O)NCC(C)(O)CNC(=O)CCc2cnc[nH]2)c(F)cccc1F 33516,C1(C(N2CC3C(NC(C4CC5COCC5C4)=O)(C3)C2)=O)CC2(C1)CC(F)(F)C2 33517,c1(CC)ccc(C=CC(=O)NCC2CCCN(C(C3CC3C(=O)OC)=O)C2)cc1 33518,C12(CCCCCCC1)C(=O)N2.c1(CC)cc(C(F)(F)F)cnc1C 33519,N1(C(c2cn(CC(C)C)nn2)C)CC(=O)N(Cc2ncnn2C)C1=O 33520,C(=O)(C(CN(C)C)NC(C1CC1(C)C(F)F)=O)NC(C)C(=O)N(C)C 33521,C1(NC(c2nc[nH]n2)C)CC(NC(=O)CNC(=O)Nc2ccco2)C12CCC2 33522,c1(CCC)nc(C(=O)N(CCCCN(C)C(C2(C)CCC2)=O)C)cs1 33523,c1(C(=O)NCC2N(C(CC(=O)OC(C)(C)C)=O)CCOC2)cc2ncccc2s1 33524,c1(NS(C)(=O)=O)cccc(NCC2COCC2C(=O)O)c1 33525,C1(C(N(C2CC(C#N)C2)CC(=O)NCC(C#C)OC)=O)CCOC1(C)C 33526,c1(CCC(C)N(C=O)Cc2cc(C(F)F)no2)ccc(C(F)(F)F)cc1 33527,C1(C(C)C)C(C(=O)NCCN2CCNC(=O)C2)CCN1C(=O)CC1CCSC1 33528,C(=O)(CCCN=[N+]=[N-])N1C2(C(=O)NC3CN(CCC)C3)CC2CC1 33529,C1(C(N2CC3(CCN(C(c4ccc([N+](=O)[O-])o4)=O)C3)C2)=O)CC2CC(O)C(C1)C2 33530,C(CCCCCN(C)C(C1CCC(CO)CC1)=O)NC(CCNC(=O)NC)=O 33531,CCCCC(CC)C(=O)N1CCC(=CCNC(C2CC3CC3C2)=O)CC1 33532,N1(C(CC(CC#C)NC(=O)CC2CCCCC2O)=O)CC(=O)NC2(CC2)C1 33533,N1(C(c2cccc(C)c2)=O)CCN(C(c2ccn(CCO)c2C)=O)C2CCC12 33534,c1(C(=O)NC2CN(C(C(CO)NC(C(C)C)=O)=O)C2)ccc2c(c1)CCN2C 33535,C1(O)(CC(=O)NCCSC)CCN(Cc2ccc(F)c(OC)c2)CC1 33536,C(=O)(CC(C)(C(F)F)N(C)C)NC(CN(C(c1ccc(C)cn1)=O)C)C 33537,Cc1cc(CC(N2CCCC2CNC(c2ccn(C)n2)=O)=O)ccc1Cl 33538,C1(NC(C2(CSC)CCC2)=O)CS(=O)(=O)CC1NC(=O)C(F)=C1CCC1 33539,c1(CC)cc(C)c(C(=O)NC2COC(C3CCNCC3)C2)o1 33540,CC12CCN(C1)C2=O.c1(C(=O)NC2(c3cccs3)CC2)ccc(NC2CC2)cc1 33541,c1(SC(C(=O)NC(CNC(c2cc(CCC)on2)=O)C)C)ccc(F)cc1 33542,C1(C(=O)NC2CN(C(=O)CC3CC(CF)C3)CC2C(F)F)SC2C=CC1CC2 33543,C(=O)(CC(C)(C(F)F)N(C)C)NC1C(O)CCN(C(CC=CC=C)=O)C1 33544,N1(C(C2N(C(C3C(CCC)C3)=O)CSC2)=O)CCCC1(C)CC1CC1 33545,N1(C2CCN(C(C3CC34CCOC4)C(=O)NCCC)CC2)CCN(CC)CC1=O 33546,C12(C(=O)Nc3cccc(C)c3)CCCN(c3ncc(F)cn3)CC1C2 33547,C1(CC#C)CN(C(=O)COC2CN(C(=O)CSC(C)C)C2)CCO1 33548,c1(CNC(c2ccco2)=O)noc(-c2cnn(-c3cnccn3)n2)n1 33549,C(C(CC(F)(F)F)NC(=O)C1=NOC(C)C1)NC(C(NOC)=O)=O 33550,c1(CNC(c2nc(CC)oc2C)=O)ccc2c(c1)CN(C(=O)CCOC)C2 33551,N1(C(C(C)OC)=O)CCC(N(CC(C)C)C(=O)C=CC2CCCCC2)CC1 33552,c1(CC)cccc(CC(=O)N(CC(CC)NC(=O)CCn2ccccc2=O)C)c1 33553,N1(C(C2N(CC)CCOC2)=O)CCCCC(NC(=O)C(c2ccccc2C)C)C1 33554,C(=O)(CCC(C)(C)N(C(N1CC=CC1)=O)C(C)C)N(CC=C)CC=C 33555,c1(SC)cncc(NC(C2(CNC(=O)C(C)NC(=O)C3CC3)CCCO2)=O)n1 33556,C1(C(=O)NCC(O)C(N)=O)(OC)CCN(C(C2CC(O)CN2C)=O)C1 33557,C(=O)(C#CC1CCCO1)NC(CNC(c1c(SCC)cccc1)=O)(C)CO 33558,N1(C(=O)NC2C(C(N)=O)CCCC2)CCOC2(CCS(=O)(=O)C2)C1 33559,Cc1cc(O)nnc1C(=O)NCC1(C)CCN(C(=O)CC2CCC(C)C2)CC1 33560,C(CC(C(=O)NC(C)CNC(c1cc(C(=O)O)n(C)n1)=O)NC(C)=O)SC 33561,C1(NC(c2[nH]c(=NC)sc2)=O)CN(C(c2ccnnc2S)=O)C2(CCCCC2)C1 33562,C1(C(=O)NCCc2ccc(Br)cc2)CC1C1CCNCC1 33563,CCCCS(=O)(=O)CC(=O)NC(C)CN(C(C1CCCN1S(C)(=O)=O)=O)CC 33564,N1(C(C2C(C)(C)NC(=O)C2)=O)CCC2(CCCN2C(C2CC(O)C2)=O)CC1 33565,N1(c2c(C)cnc(Cl)n2)CC(NC(C2CC3(C2)CC(O)C3)=O)CC(C)(C)C1 33566,N1(C(C)=O)CCC12CN(C(c1oc(-c3ccccc3)cc1C)=O)C2 33567,Cc1cc(C(C)(C)NC(=O)NCC2CC(F)(F)C2)cc(C)c1Cl 33568,Cc1ccc(C)c(OCC(N2CC(O)(CNC(c3csc([N+](=O)[O-])c3)=O)C2)=O)c1 33569,C1(CC(=O)OC)CN(C(=O)CC(=O)N(C)C)CC1C.c12cn(nn1)NC2 33570,Cc1ncc(C(F)(F)F)cc1C(=O)NC1CC(NC(=O)C=Cc2ccc[nH]2)C1 33571,c1(CNC(C=CCC2(NC(c3c(CC)ocn3)=O)CCC2)=O)oc(C)nc1C 33572,c1(C(N2CC(CCNC(c3c(CC)nns3)=O)(OC)C2)=O)cc(C(C)C)nn1C 33573,c1(NC(=O)OC2CCC2)cc(OCC(N2CCC(O)C2)C)ccn1 33574,CCC(C(=O)NC(CCSC)C(=O)NCC1(C#N)CCCCC1)C(F)(F)F 33575,N1(C(c2cnn(C)n2)=O)CCN(C2CN(C(C3CCCC3C(F)F)=O)C2)CC1 33576,Cc1nc(C(=O)NC2CC(CCC(=O)NCC3(N(C)C)CC3)C2)c(C)o1 33577,C1(CN(C(=O)Cn2cnnc2)C)CCC(CNC(=O)C=CCn2cncn2)CC1 33578,Cc1nn(C2CCOCC2)cc1C(=O)NCC1(NC(=O)C=CS(C)=O)CCCC1 33579,c1(CN2CC3CCC(CC(=O)OC)(C2)C3)cc(F)cc(F)c1Br 33580,CCCCCC(=O)NC12COC(CNC(C3(C)CCC(=O)N3)=O)(C1)C2 33581,N1(C(C=Cc2cn(C)nn2)=O)CCN(C(c2ccsc2C#N)=O)CC(CO)C1 33582,c1(OC)cc(S(=O)(=O)ON2CCCC2)ccc1N(C)C 33583,C(=O)(C(C)C(F)(F)F)N1CCC(CCNC(c2cccc(C)n2)=O)CC1 33584,C1(NC(C=CC=CC)=O)CCCC12CN(C(c1cccc(C(F)(F)F)n1)=O)C2 33585,c1(C(=O)NC2(C)CCCN(C(c3cc(C)on3)=O)C2)cc2cnccc2o1 33586,c1(OC)c(C(=O)OC(C)C(C)n2cccn2)oc2ccccc12 33587,C(CCCOC)(C(=O)N1CC(C(C)C)C1)NC(c1nn(CC)nc1C)=O 33588,c1(C(N(C)CC2CCN(C(c3ccc(C(F)F)s3)=O)C2)=O)cc2cnccc2o1 33589,N(C(=NCCCCl)NCc1nnnn1-c1ccccc1Cl)CC1CC(=O)NC1 33590,C1(C(C)N(CC(CF)C2(O)CCC2)CCO)CCOC1 33591,N1(C(C(N2CCC(C)C2)=O)=O)CCC(O)(CSc2ccccc2)CC1 33592,C1(NC(C(=O)NCC)=O)(CO)CCCN(C(c2ccccc2Cl)=O)C1 33593,c1(C(=O)OCC)nc(=NC2CC(F)(CNC(=O)CN(C)C)C2)cc[nH]1 33594,Cc1c(Cl)cc(C(=O)NCCCC(=O)N(CCCN)C)cc1I 33595,CCC(C(=O)N1CC(N(C)C(c2csc(C)c2OC)=O)C1)C(C)C 33596,C1(CC)CN(C(=O)CCCC(N)=O)CCN1C(=O)C(CC)OC 33597,C1(C(=O)NCC2CCC(NC(=O)CCCC3OCCO3)C2)C2CCC1CC2 33598,C#CC1(NC(=O)CCCC(C)NC(c2coc(C(N)=O)c2)=O)CCCCC1 33599,C1(NC(c2ccccc2-c2nc[nH]n2)=O)CN(C(C2CC2(F)F)=O)CC1C(F)F 33600,C(=O)(C1=C(Cl)CCCC1)N1C(CN(C(C2(SCC)CC2)=O)C)CC(F)C1 33601,C1(NC(c2nc(C(C)NC(CC(C)C)=O)oc2)=O)CCN2CCC1C2 33602,C(CC(O)CCC(C)(C)C)NCCc1cn(CCOC)nn1 33603,CCC(C)C(C(=O)NCC1COCCN1C)N(C(=O)CCC(C)OC)C 33604,N1(C(=O)Cc2ccon2)CC2CC(NC(=O)C(F)(F)Cc3ccc(F)cc3)C1C2 33605,C1(CNC(C(CCOC)C)=O)CCC2(CN(C(C3CCOC(C)C3)=O)C2)O1 33606,C(=O)(CCc1ccc[nH]1)N(C(C)C(=O)NC(C)C(=O)NC)CC 33607,CN=c1cc(C(=O)NC2CCC(CCNC(=O)Cn3nnc(=O)[nH]3)C2)cc[nH]1 33608,c1(N(C)C)ccc(C(=O)NC2CN(C(C3(C)CCC(=O)C3)=O)CC2F)cc1 33609,N1(C2CN(C(c3cnc(C)s3)=O)C2)CCN(C(c2cc(C(F)F)on2)=O)CC1=O 33610,C#Cc1ccc(C)c(NC(=O)C(CCC=C)NC(c2sncc2C)=O)c1 33611,Cc1cc(-n2cc(C3CCC(C)CC3)nn2)cc(=O)o1.c12ccc(c(C)c1)o2 33612,CC(C)(CS(N)(=O)=O)C(=O)N1CCN(C(C2CCC3(CC2)CC3)=O)CC12CC2 33613,C(C(CC(C)C)C(=O)NCC1C(CC)CCN1C(c1ccc(CO)cn1)=O)OC 33614,C=CC(C(=O)N(C1CCN(C(c2cnccn2)=O)C1)CC)NC(=O)OC(C)(C)C 33615,C(N=c1nnc(C)c(C)[nH]1)C1C(NC(c2ccc(C)c(F)c2)=O)CCC1 33616,N1(CC(=O)NCC(CC(C)C)NC(C2CCC23CCC3)=O)CCc2sccc2C1 33617,N1(C(c2cc(C(C)=O)sc2)=O)CCN(C(=O)C(F)(F)c2cccnc2)CC1CF 33618,c1(NCCC(=O)NC)nc(=NCC(C(C)C)N(C)C)[nH]c2c(C)nn(C)c12 33619,c1(C(C(=O)NCCN(C(=O)C(C)C(C)C)CC)(C)O)cccc(Br)c1 33620,C(CC(C)C(=O)NCCCC)=CC.C1CCN(C(C2(n3cc(Cl)cn3)CC2)=O)C1 33621,C1(C(=O)NCC(C)NC(c2cc(Cl)ncc2N)=O)CCc2cc(F)ccc2O1 33622,CC1CC(NC(=O)Cc2ccc(F)cc2)CN1C(=O)CC1CCS(=O)(=O)C1 33623,CCCC(CCCNC(c1cc(Br)nn1C)=O)Nc1ncc(C)cn1 33624,Cc1cccc(C)c1NC(=O)C(c1cc(Br)ncc1F)N1CCC(C(F)F)CC1 33625,C(=O)(CC(CC)CCC)NCC1CCCN(C(C(C#C)(C)C)=O)C1 33626,CC(C)CCC(F)C(=O)NC1CC1CNC(c1cc(C(N)=O)n(C)n1)=O 33627,c1(SCC(=O)NCCC2CCCN(C(C=C(C)C)=O)C2)nc2ccccc2s1 33628,Nc1nc(C(N2CC(NC(c3cnns3)=O)CC(O)C2)=O)cnc1Br 33629,C(=O)(C(C)(F)CCCC)NC(CC(=O)NCCCC(C=C)(C)C)CCC 33630,c1(CN(CC(C)C)N(C)C(C)c2nncn2C)nnc2n1CCOCC2 33631,c1(C(N2CC3(CC3C(N3CCC(c4cn[nH]c4)CC3)=O)C2)=O)cccc(Cl)c1Cl 33632,c1(C(=O)NCC(CC(C)C)NC(C(C(CC)(C)C)O)=O)c(C)nc2ccccn12 33633,C1(CNC(C2CCCN(C(C)=O)C2)=O)CCCCN(C(C23CC(C2)C(C)O3)=O)C1 33634,CCCC(CC)C(=O)N1CC2C(CNC(=O)C(CC)n3ccnc3)C2C1 33635,N1(C(c2nc(CCC)sc2)=O)CC(CNC(=O)C=CC2CC2)C2CC12 33636,Cc1cccc(-c2cccnc2NCC(N2CCN(C)CC2)=O)c1C 33637,N1(C(CCCNC(C)=O)=O)CCN(C2CCCN(C(=O)C(O)C(F)F)C2)CC1 33638,CC1(C)CC(C(N2CCOC(CF)C2)=O)CCN1C(=O)CCc1nncs1 33639,C1(NC(C(C)CC(F)(F)F)=O)C2CC3CN(C(=O)C4=COCCO4)C1C3C2 33640,CC1CCN(C(=O)C(=O)NCC(C)Cc2cnn(C)c2)CCS1 33641,c1(NC(C2C(C)CCCC2)=O)cnc2ccc(F)cc2c1 33642,CC1CCN(C(c2cc(O)nn2C)=O)C1CNC(c1ccc(C2(C)CC2)cc1)=O 33643,c1(C(C)(CO)N(C(=O)NCC2CCN(C)C2)Cc2ccco2)cccc(C(F)(F)F)c1 33644,c1(NCCC2(COC)CC2)ncnc(N(C(CO)CC(C)C)C)c1C 33645,C1(O)(COC)CN(C(=O)C(F)CC2CN(C(=O)C(c3ccc(C)o3)C)C2)C1 33646,c1(C(N(CC)CC2CCCN(C(=O)CC(C)(C)SC)C2)=O)cnc(C)c(N)c1 33647,Cc1cnc(C(N2CCC(CO)(NC(=O)OC(C)(C)C)C2)=O)cc1C 33648,C1(C(=O)NC2COCCN(C(CN3CCC(C)(C)C3)=O)C2)CCCC2(CCC2)O1 33649,Cc1cc(F)cc(C)c1C(=O)NC1CCN(C(c2[nH]cnc2C#N)=O)C1 33650,c1(CN2CC=CC(OC)C2)nc2ccc(Br)nc2[nH]1 33651,N1(C(c2nc(CC)oc2C)=O)CC(NC(c2cnc(C)c(C)c2)=O)CC12CCC2 33652,Cc1cc(C(C)NC(=O)C(=O)NC(c2ccccn2)C)on1 33653,c1(C(N(CC(CO)(CO)NC(C2C(C)C2C)=O)C)=O)n[nH]c2c1CCCC2 33654,C1(C(=O)NCC23C(CN(C(C=CC(N)=O)=O)C2)C3)COc2ccccc2O1 33655,C#Cc1ccc(C(=O)NC2(COC)CCN(C(=O)C(C(C)C)NS(C)(=O)=O)C2)nc1 33656,C=CCCCC(=O)NCC(CC=C)NC(=O)C(=C1CCCCC1)F 33657,c1(C(=O)NCC(C)CNC(C2CCN(C)C2)=O)oc2ccccc2c1CO 33658,N1(C(c2nc(CC)oc2C)=O)CCC2CN(C(c3cn(C)nc3OC)=O)CC12 33659,C=C(C)CCC(=O)NCC(CO)NC(=O)CC(C)C 33660,C(=O)(C(C(C)O)NC(=O)Cc1cn[nH]c1)NCC1(C(C)C)CCCC1 33661,C1(C(=O)Nc2ncc(S(C)(=O)=O)s2)CCCC12CCCCC2 33662,C(=O)(C1=CCCCO1)N1CCN(C2CCCN(C(CSC)=O)C2)CC1 33663,c1(C(=O)NC2C(C)N(C(=O)Cn3ncnn3)CC2)cc2c([nH]1)CCOC2 33664,CC(C)(CCC(=O)NC1CCC(C(N)=O)C1)NC(C1CC=CC(O)C1)=O 33665,CCCCC(N)C(=O)NCc1ccc(F)nc1F 33666,Cc1nncc(C(N2CCCC2C(C)NC(C2CC23CCC3)=O)=O)c1C 33667,C(C)(CNC(C1CCNC1=O)=O)(CO)NC(C(C)=CC1CC1)=O 33668,C1(OC)CCCCCC1Nc1ccc(-c2ccc(C)nc2O)cn1 33669,c1(C(N2CCC(NC(C3N(CC)CCC3)=O)C2)=O)nc2ccc(C)cn2c1N 33670,C(CC(C)(C)N(C1CCC1)C(c1ccncn1)=O)N(C1(C(=O)N(C)C)CC1)C 33671,c1(C(=O)NCC2C(NC(c3c(OC)cccc3)=O)CCC2)ccc(C)c(C)c1 33672,C=CC(CC)CC(=O)N(C1CCCN(C(=O)C(O)C2CC2)C1)CC 33673,c1(C2(NC(CCc3nnc(C)o3)=O)CCCC2)ccc(OCc2cccs2)cc1 33674,CC1(C(=O)NCC2CC(NC(=O)CCc3cnoc3)C2)CC(C#N)C1 33675,c1(OC)ccc(NCc2cc(C)c(-c3ccc(C(C)O)cc3)s2)cc1C 33676,C1(N(C)C)(C(=O)NCC(O)CCNC(=O)CCC2CCC2)CCOCC1 33677,C12(NC(C3CCOC3)=O)CCC(C1)N(C(c1cc(Cl)ccc1-n1cccc1)=O)C2 33678,c1(C(=O)O)cc(C(=O)N(CCn2cc(CC3(O)COC3)nn2)CC2CC2)ccn1 33679,C1(OCC)CCC1C(=O)N(C1(C(=O)N(CCCO)C2CCC2)CC1)C 33680,C(C(=O)NCc1cccs1)(C(C(C)C)OC)N1CCCC(C(=O)OC)C1 33681,C(=O)(C1=NOC2(C1)CN(C(=O)OC(C)(C)C)C2)N(CCO)CC=C(C)C1CC1 33682,c1(N(C)Cc2ccoc2)ccc(S(=O)(=O)NC2CC3CCC(C2)S3)cc1F 33683,c1(C(=O)NCCCN(C(C(CSC)O)=O)C)ccc2c(c1)CC(=O)NC2 33684,C=CC(C)(O)CC(=O)N(CCC(C(C)(C)C)NC(=O)CCOCC(F)F)C 33685,C1(NC(C(C(=C)Cl)(C)C)=O)CN(C(=O)C(C)CC(=C)C)C2(CCC2)C1 33686,C1(CNC(C(C)Sc2nncn2C)=O)CCCC(NC(=O)CCn2cccn2)C1 33687,N1(CC)CC(C(N2CC3CC2C3NC(=O)CSc2n[nH]c(C)n2)=O)CCC1=O 33688,N1(CC)CCCCC1C(=O)N(C1CCN(C(=O)CCSc2ccccc2C)C1)C 33689,c1(C(=O)NCCC23C(CN(C(CCOCC)=O)C2)CC3)sc2ccccc2c1C 33690,c1(C(=O)NCC(C)CNC(=O)CCn2cc(Cl)cn2)ccc([N+](=O)[O-])c(O)c1 33691,c1(N2CCC(NC(C3(C)ON=C(C)C3)=O)C2)nc(C)c(C#N)cc1Cl 33692,c1(C2(SCC(=O)Nc3cncc(C(=O)OC)c3)CC2)ccc2c(c1)OCCCO2 33693,N1(C(c2ccn(C(C)C)n2)=O)CCCC2(NC(=O)C(C)n3ccnc3)CC2C1 33694,c1(C(=O)NC(CCN(C(C(CSC)OC)=O)C)C)c[nH]cc(Br)c1=O 33695,N1(C(c2nc(C)n(C)c2)=O)CCCC(NC(c2[nH]ncc2C#N)=O)CC1 33696,CCCC(CC)C(=O)NC1CCC(NC(c2ccc(C)cn2)=O)C1 33697,N1(C(c2ccc(OC)o2)=O)CC(NC(C2CCS(=O)CC2)=O)C(O)C1 33698,N1(C(C(c2ccc(OC)cc2)C)=O)CC(C2CCN(C(=O)C(O)C3CC3)CC2)C1 33699,c1(C(CC)NC(=O)CCCc2ccc(C)nc2)cc(C)ccc1OC 33700,CC(C)(C)C(C(=O)NC12CC(NC(c3csc(=N)[nH]3)=O)(C1)C2)N1CCCC1=O 33701,CC1CN(C(C2CCCN2C)=O)CC(C)CN1C(=O)CCc1ccco1 33702,CNS(=O)(=O)NCC(=O)NCC1CC1NC(C1CCOC1C)=O 33703,c1(NC(CCC)=O)ccnc(C(N2CC(CO)(NC(C3CCC4CC34)=O)C2)=O)c1 33704,C1(CCC(=O)NC(CNC(C(C)=C(CC)C)=O)CC)CCC(=O)NC1 33705,C1(C(=O)NCC2(COC)CN(C(C(C=C)C)=O)C2)CCC2(CCC2)C1 33706,C(=O)(C(O)CC(C)(C)C)N1CCC(N(C)C(c2cc(-n3cnnc3)ccn2)=O)C1 33707,N1(C(C2(CNC(c3cc(C)sn3)=O)CCC2)=O)CC(C)(C)OC(C)(C)C1 33708,Cc1cnc2c(C(=O)NCC(C)NC(C3CC34CCCCC4)=O)cnn2c1 33709,CS(=O)C=CC(=O)NCC1C2CN(C(C3CC(O)(c4cccnc4)C3)=O)CC12 33710,c1(C(N2C(C3CCN(C(C=C(COC)C)=O)C3)CCC2)=O)ccc(N)cc1C 33711,CC1Cc2cccc(C(=O)N(C(CNC(c3ncc[nH]c3=O)=O)C3CC3)C)c2O1 33712,c1(-c2nc(Cc3c(OC)ccc(Br)c3)nn2CCF)cncc2nc[nH]c12 33713,c1(C(=O)NCCSCC(=O)O)ccc(-n2cc(-c3cncc(CO)c3)nn2)cc1 33714,c1(CNC(N(C(C(=O)OCC)C)C)=O)ncncc1C 33715,C1(C(=O)NCC2CCCC2CF)(NC(=O)COC2CCCC2)CC(F)(F)C1 33716,S(=O)(=O)(c1cnn2ncccc12)N1CC(OC(C)(C)C)C(C(=O)NC2CC2)CC1 33717,C(c1cccc(F)c1Cl)=CC(=O)NCCCCCNC(Cc1cn(C)nn1)=O 33718,c1(C(=O)NCC(CCOC)NC(c2csnc2OC)=O)cc(C)ccc1C 33719,c1(C(N2CC3(C(NC(CCCOCCOC)=O)CC3)C2)=O)cnc2c[nH]nc2c1 33720,C1(O)(C(C)NC(=O)CC(C)n2cccn2)CCN(C(=O)CC(C)N(C)C)C1 33721,CCCC(CCCNC(=O)CC1COCC1(C)C)NC(c1cnc[nH]1)=O 33722,C1(NC(C(CC)CC)=O)CCC(C)N(C(=O)C(c2cccc(Br)c2)C)C1 33723,c1(OC)c(C(=O)NC2COCC2NC(=O)Cn2nc(C)nc2C)ncnc1C 33724,Cc1cccc(Br)c1C(C(=O)NC1CC1c1ccco1)NC(c1nn(C)cc1C)=O 33725,c1(N2CCN(C(C34CNCC3(F)CCOC4)=O)CC2)ccc2c(c1)C1(CC1)C(=O)N2 33726,Cc1cccc2c1OCCN(C(=O)C(C)(N)CC(C)C)C2 33727,CCCS(=O)(=O)C(C)C(=O)NCC1CC2(C1)CN(C(C1CC1(C)C)=O)C2 33728,C1(C(N2CCC(N(C(COCCC#C)=O)CCO)CC2)=O)CC2(C1)CC1(CC1)C2 33729,c1(C(=O)NC(CNC(c2cncc(CC)c2)=O)CO)cc(C(C)C)ccc1N 33730,c1(C(N2CCC(C(O)CO)C2)C(=O)NCCCC2CC2)ncc(Cl)s1 33731,N1(C(C2C(CC)OCC2)=O)CCC(F)(CNC(C23CC2C3)=O)CC1 33732,CC(CC(F)(F)F)C(=O)NCCNC(C1CCCN(C(=O)C#CC2CCC2)C1)=O 33733,C=CC1(C(=O)N(C2C3CCCC23)C)CCN(C(c2cccnn2)=O)C1 33734,C1(NC(C(C2CC2)OCC)=O)CCCCCC1NC(c1ccc(N)c(SC)c1)=O 33735,C1(COC)(CNC(=O)COC(C)C)CCN(C(=O)CNc2ccncc2)CC1 33736,c1(C(=O)NC(c2cccnc2)C(=O)NCC2(OC)CC2)cnc(C2CC2)o1 33737,Cc1ncc(C(=O)NCC2CCC(NC(=O)Cc3c(C)ncnc3O)C2)cc1N 33738,c1(NC)ccc(C(F)(F)F)cc1C(=O)NC1CN(C(C2COC(=O)N2)=O)C1 33739,C(=O)(N=c1cc2ccccn2[nH]1)C1(C)C=CCN1C(c1cc(Cl)cs1)=O 33740,c1(OC(C)(C)C)ccc(C(=O)NC2CCN(C(c3coc(Br)n3)=O)CC2)cn1 33741,c1(C(N(CC(C)NC(=O)CC#N)C)=O)cnoc1C1CCOCC1 33742,N1(C(CSC(C)(C)C)=O)CCN(C(=O)C(F)C(C)(F)F)CC1c1cn[nH]c1 33743,Cc1cc(C(=O)NCC(C)(CO)NC(=O)CCc2cc(Cl)no2)ccc1Cl 33744,C1(CCNC(=O)CCCn2cncn2)(OC)CN(C(=O)C(c2ccc(C)s2)C)C1 33745,O=C1CCc2c(C(=O)Nc3cc(Cl)c(Br)c(Cl)c3)cccc21 33746,c1(C(c2ccco2)=O)nn2c(c1CNCC(O)COc1ccc(Cl)cc1)CCC2 33747,c1(CNC(=O)C(N2CC(CO)C(c3ccccc3)C2)=O)c(F)cncc1F 33748,CN1C(=O)CCC(c2nc(C3(c4ccccc4F)CC3)no2)C1c1cccc(Cl)c1 33749,N1(C(COCC(C)C)=O)CCC(C)(CCNC(C2CC(C)C2)=O)C1 33750,Cc1nn(C)c(C)c1C(N1CC2CC1(CNC(C1(CO)CCCCC1)=O)C2)=O 33751,C1(CCNC(c2cc(C)on2)=O)CCN(C(C2CCCN2C=O)=O)CC1(F)F 33752,C12C(C1(C)C)C(=O)N2.C1(CCNC(C2CC(N(C)C)C2)=O)CC(F)(F)C1 33753,N1(C(C2C=C(C)CS2)=O)CC(CC(N2CCCC(F)(CO)C2)=O)C2(CC2)C1 33754,Cc1ccoc1CNC(=O)CN(C(C1CC1F)=O)CC1CC1 33755,C1(CC)CN(C(C2(NC(=O)CC(C)CN(C)C)CCOCC2)=O)CC(=O)N1 33756,c1(CSC)cccnc1C(N1CCOC(CNC(C2CCC(=O)N2C)=O)C1)=O 33757,S(=O)(=O)(c1cccnc1N1CSC(C)C1)N(C(C)=O)CC1CCCOC1C(C)(C)C 33758,CCCCC(F)C(=O)N(C1CCCN(C(c2c[nH]c(=N)c(C)c2)=O)C1)CC1CC1 33759,CCC(C)(C)C(=O)C(=O)N1CC(F)(C(=O)NC2(C(C)O)CC2)C1 33760,c1(C(=O)NC2C(CNC(c3c(CC)c[nH]c3)=O)CCCC2)cn(C)c(=O)cn1 33761,c1(C(N(C(CNC(C2CCC(=O)O2)=O)C2CC2)C)=O)cc2ccccn2n1 33762,N1(C(C2CC(C)SCC2)=O)CCC(C)(C)C1C(=O)NCCCSC(F)F 33763,c1(CC)cccc(N(C)C(c2cc(CNC(=O)CC3CC=CCC3)no2)=O)c1 33764,C(=O)(C(S(C)(=O)=O)C1CC1)N(C(C)CNC(c1ccc(Cl)o1)=O)CC 33765,C1(OC)CCCC(CNC(=O)CN(C(=O)Cn2cncn2)CC2CC2)C1 33766,C1(C2CCCC2)(C(=O)NC2C3(CCN(C(c4cc(Cl)nnc4O)=O)C3)C2)CCC1 33767,C(=O)(C(O)C(F)(F)F)N1CC(O)(CNC(c2ccc(CC)s2)=O)C1 33768,CC1COCCCN1C(C1CC1C(C)NC(=O)Cc1ccccc1O)=O 33769,Nc1cnc(Cl)c(C(N2CCOCC(NC(c3ccc(F)s3)=O)C2)=O)c1 33770,c1(CC(=O)N(CCCNC(c2ncn(CC)c2)=O)C2CC2)cccc(OC)c1 33771,c1(C(N2CCC(CN(C)C(C3CCCN3C=O)=O)CC2)=O)cc(O)c(O)c(O)c1 33772,Cc1ccc(Br)cc1C(N1CCC(CO)C(C)C1)C(=O)NCCCF 33773,C1(c2n(CC(F)F)nnn2)(NCC23COC(CF)(C2)C3)CCN2CCCCC2C1 33774,C1(CNC(C2(CC)CCN(C(C3CCCSC3)=O)C2)=O)CCC(C)(C)CC1 33775,c1(CC(=O)NCC(CC)(C)NC(=O)CCC2CC(F)(F)C2)ccc(Cl)c(C)c1 33776,N1(C(CCC(=C)C)=O)CCN(C(=O)C(C)CCC)C(c2cn[nH]c2)C1 33777,c1(C(N(CC(C)(C)NC(CNC(=O)OCC=C)=O)C)=O)cnc(CCOCC)[nH]1 33778,c1(C(=O)NCC2CN(C(=O)CCc3cncs3)C2)cccc2cncn12 33779,C#Cc1cc(C(=O)NCCNC(C2CC[Si](C)(C)CC2)=O)cc(F)c1 33780,N(C(=NCCOc1ncccn1)NC1CC(CNS(C)(=O)=O)C1)CCSCC=C 33781,C1(c2nn(CCC)c(-c3ccc(C)nc3)n2)CCC(F)(F)CC1 33782,c1(CNC(C2N(CC)CCC2)=O)sc(OC)nc1Cl 33783,c1(CCc2c(OC)ccc(OC)c2)nc(C)nc2scc(CCO)c12 33784,C1(NC(CNC(C)=O)=O)COCCC1NC(c1cccnc1-n1nccn1)=O 33785,c1(CC(=O)NCC2C(NC(CNC(=O)OC(C)(C)C)=O)CC2)ccc(Cl)o1 33786,C=C1CCN(C(c2nscc2C)=O)C(C(=O)NCCC2CC=CCC2)C1 33787,Cc1ccc(C(=O)NC(C)C(CO)NC(c2cc(C(=O)OC)sc2C)=O)c(O)n1 33788,c1(C(=O)NCC2(F)CN(C(CSCCCC)=O)C2)cccc(C(=O)NC)c1 33789,c1(C(N(C(CNC(CC=C)=O)C)CC)=O)cnc(Br)c(N)n1 33790,N1(C(C2C(C(N(CCCO)C)=O)CC2)=O)CC2(CNC(=O)C2)C1 33791,c1(CC(=O)N(CCn2cc(CC(O)CO)nn2)CC)cc(Cl)cc2c1OCC2 33792,CC1(C)OCCOC1C(=O)NCC1(O)CN(C(c2ncsc2C2CC2)=O)C1 33793,N1(C(c2ccc(C)[nH]2)=O)CCN(C)C(CNC(=O)C(c2cccnc2)O)C1 33794,N1(C(C(C)=CC)=O)CC(C)(C)CC1CNC(=O)CC(=O)N(C)C 33795,C1(CNC(C(C(C)C)C)=O)CN(C(c2cnc(Cl)c(N)c2)=O)C2COCC2O1 33796,C1(C)(OC)CCCN(C(=O)C(C)(CNC(c2ncoc2C)=O)CC)C1 33797,CN1CCOCC1C(=O)N(C)Cc1ccc(CNC(=O)CN(C)C2CC2)cc1 33798,CCC(CC(C)C)C(=O)NCCN(c1ncc([N+](=O)[O-])cn1)CCOC 33799,N1(C(C(C(CC)C)OC)=O)CC2CCC(C1)N2C(=O)C(N1CCN(C)CC1)(C)C 33800,c1(C(N2CC(Cn3cc(CCNC(C)=O)nn3)C2)=O)cc(F)cnc1O 33801,C(=O)(C(CC(C)C)NC(c1c[nH]c(C#N)c1)=O)NC(C(CC)CC)C 33802,C1(C(=O)NCC2C(C)CN2C(=O)C2=COCC2)CCC(C2CCC2)CC1 33803,C1(CC(=O)NCC(CNC(=O)CCc2nccs2)F)CCCCC12CC2 33804,N1(C(C(CC)c2ccccc2)=O)CC(CNC(=O)CC(C)(F)F)C2(CC2)C1 33805,c1(CNC(C2C(CNC(C(CN(C)C)N(C)C)=O)C2(C)C)=O)cccc(O)c1 33806,c1(C(=O)NC2CCCC(NC(CNC(=O)NC)=O)C2)cc(C)cc(F)c1 33807,c1(CNC(C2(CC(C)C)CC2)=O)ccc(CN(C)C(C2C(F)(F)C23CC3)=O)cc1 33808,c1(C(N2CCCC(CNC(=O)NC)C2)=O)cc(C#N)c(Br)s1 33809,CC1CCN(C(=O)OC(C)(C)C)C1C(=O)NCC1CCC(CC(F)(F)F)CC1 33810,N1(C(c2ccc(C)cc2)=O)CCC(N(C)C(C23CC4CC2C3C4)=O)C(C)C1 33811,C1(COC)(CNC(=O)Cc2c[nH]nc2O)CCCN1C(C1CNC(=O)N1)=O 33812,c1(OC)c[nH]nc1C(N1CC(CNC(=O)CCC2CCCCC2)(OC)C1)=O 33813,c1(CC)ccc(C(N2CC(NC(C3(OC)CCCC3)=O)C3CC23)=O)c(OC)c1 33814,Cc1ccc(CCC(N2CC(C)(NC(c3cc(Cl)c(Cl)[nH]3)=O)C2)=O)cc1Cl 33815,C(CCC(C)NC(=O)CN1CCOC1=O)NC(C(C)SCC)=O 33816,Cc1nnc2n1C(C(=O)N1CCN(C(c3csc4nnsc34)=O)C(C)C1)CC2 33817,N#Cc1cnn(CC(=O)OCCOc2ccc(Cl)cc2)c1 33818,FCCN=C(NCCNc1ccccn1)N1CCCC2(CCCNC2=O)C1 33819,C1(CNC(C2N(C)C(=O)NC2)=O)C(O)C(O)CN1C(c1ccc(F)cc1)=O 33820,c1(CC(N2CC3(CCN3C(c3ccc[nH]3)=O)C2)=O)cc(Cl)cc(Cl)c1 33821,O=C(C1=CCCC1)N1CCCC1CCCNC(C12CC(CN1C1CC1)C2)=O 33822,C1(CC(N2CCC(NC(=O)CC3CC=CC3)(CF)C2)=O)CN2CCN1CC2 33823,C=CCCC(C(=O)Nc1ccc(C)nc1)NC(c1cc(C)n(CC)n1)=O 33824,N1(C(c2ncc(OCC)nc2)=O)CCCC(N(C)C(c2csc(C)c2N)=O)CC1 33825,Cc1cccc(C(N2C(C(=O)NCC=Cc3cccnc3)CCC2CO)=O)c1F 33826,c1(CN2CCC(N(C(C=CC(C)C)=O)C)CC2)ccc([N+](=O)[O-])cc1O 33827,C(CCCC(=O)NC1(C)CCN(C(=O)C(C)(C)c2cccnc2)C1)OCCC=C 33828,c1(C(N(CC(C)NC(CC(=C)Br)=O)C)=O)ncccc1S(=O)(=O)CC 33829,N1(C(c2cncc(COC)c2)=O)CCC2(CC1)CC2NC(C1CC2C=CC1C2)=O 33830,c1(N2CC(C)(C)C(NC(=O)CN3C(=O)CCC3=O)C2)nc2c(F)cc(Cl)cc2s1 33831,N1(C(c2c(CC)con2)=O)CCC(NC(=O)CCCN(C)C)C1c1ccccc1 33832,Cc1ccc(C#N)cc1NC(=O)C(C)N(C(=O)CSc1nc[nH]n1)C1CC1 33833,C(CC(C)C(=O)NCC1CC1NC(c1ccnnc1C)=O)=CCC 33834,Cc1cc(Cl)c(Cl)cc1C(=O)NCCN(C(=O)CC1(C)CC1F)C(C)C 33835,N1(C(c2cc(CCCCC)[nH]n2)=O)CCCOC(CNC(=O)C=CC=C(Cl)Cl)C1 33836,C1(C)(C(=O)NCC(C(=O)N2C(CC(C)C)CC2)CC2CCCC2)CC(=O)N(C)C1 33837,C1(C(C)C)CNC(=O)CN1C(C1CCC(NC(=O)COC2CCCCC2)CC1)=O 33838,C(CC(CC)C(=O)N1C(CC(=O)NCc2cn(CC)nn2)C2CCCC12)=CC 33839,C1(CC(N2CCC(O)(CN(C(=O)CSCCC#N)C)C2)=O)CC2CCC(C1)N2C 33840,N1(C(C2(C(C)=O)CC2)=O)CC2(CCN(C(=O)Cc3nnc(C)o3)C2)C1 33841,C12(CNC(Cc3nnc(C)s3)=O)CC(NC(C3CC(C)(C)C3)=O)(C1)C(C)(C)O2 33842,c1(OC)ccc(C(F)(F)C(N2CC3CC3(CNC(=O)C(C)C3CCC3)C2)=O)cc1 33843,O=C(C1=NOC2(CCN(S(=O)(=O)C3CCCC3)C2)C1)N1CCc2ncncc2C1 33844,C#CC1CCCCN1C(=O)C(c1cn(C)nn1)NC(C1CCS1(=O)=O)=O 33845,CCC(CC(=O)N1CC(CO)(NC(=O)CS(=O)(=O)NC)C1)CC(F)(F)F 33846,C1(CC)(CO)CCN(C(C2CCN(C(c3coc(SC)c3)=O)C2(C)C)=O)CC1 33847,C1(CC(N2CCC(NC(COCCN(C)C)=O)(CO)C2)=O)CC2CCC1CC2 33848,c1(C(N(CCCNC(=O)C2=NNC(=O)CC2)C)=O)ccc2nc(Br)nn2c1 33849,S(=O)(=O)(c1cc(C(=O)NC(C2CCN(C(=O)C3=COCCC3)C2)(C)C)co1)NC 33850,N1(C(C(C)OCCCC)=O)CC2CC2(C(=O)NC2CC3CCC2O3)C1 33851,C1(NC(c2c(C)cc(F)cc2)=O)CC2CC(NC(=O)C(C)(C)C3CCC3)CC2C1 33852,c12[nH]c3ccccc3c1CC1(CC)COCC(CCCNC2=O)CNC1=O 33853,N1(C(C(Cc2ccccc2)OCC)C(=O)NCCOC)CCC(S(N)(=O)=O)C1 33854,c1(OC)cc([N+](=O)[O-])cc(CN2Cc3[nH]nc(C(N)=O)c3C2)c1O 33855,C1(C)(CC)CC(NC(=O)CC2(NC(=O)C(c3cccnc3)O)CC2)C1 33856,CCC(O)(CC)CCN=C(NCc1ccc(C(N)=O)o1)NC(C)C 33857,N1(C(C2(CC=C)CCCC2)=O)CCOCC(NC(=O)CC2CCOCC2OC)C1 33858,c1(C(=O)NCC2(COC)CN(C(CNC(CC)=O)=O)C2)cc(Cl)c(OC)cc1Cl 33859,C1(CNC(Cc2c(C)nn(C)c2C)=O)CCC2(CCC2)C1NC(=O)CCF 33860,c1(C(=O)NC2CC(CNC(c3sccc3Cl)=O)C2)ncc(Cl)nc1Cl 33861,Cc1c(I)c(C(=O)OCc2cc(C3CC3)on2)nn1C 33862,O=C(CCS(=O)(=O)N1CCOCC1)N1C2CC2C2CC12 33863,Cc1cc(C(=O)N(CCCNC(=O)CC(=O)NC2CC2)CC2CC2)ccc1O 33864,C(C)(C(CO)NC(c1ncoc1CCC(F)(F)F)=O)NC(C(C)N(C)C)=O 33865,c1(C(=O)OCC)cc(NC(N2CCC(OC(C)=O)CC2)=O)ccc1C 33866,c1(OCCC(=O)NC(C(=O)NCC#C)C)c(C)ccc(C)c1C 33867,c1(C(N2CCN(C(C(C(CC)C)O)=O)C3C2CC3)=O)cnc2c(c1)CCC(=O)N2 33868,CC1CCN(C(=O)C=C(Cl)Cl)C1C(=O)NCc1ccc(Sc2nc[nH]n2)o1 33869,N1(C(CCSC)=O)CC2CC3CC2C1C3NC(c1cc2sc(C)cc2[nH]1)=O 33870,CC1CCC(c2cn(CC(C3CCCCN3)(C)C)nn2)CC1 33871,c1(C(N(CC)CC2CCOC2)=O)n[nH]cc1CNC(=O)C(C)=CC1CC1 33872,C(=O)(C(F)CC(C)(C)NC(=O)CCC1CCOCC1)N(C)Cc1nccs1 33873,Cc1ccc(C=CCNC(C)CCCc2cccnc2)cn1 33874,Cc1c(N)ccc(C(=O)NCCN(C(c2csc(Cl)n2)=O)CC2CC2)c1C 33875,N12CC3CC1CN3C2=O.C1(NC(c2nc(CC)sc2)C)CCCN(C(N)=O)C1 33876,N1(C(C(CCC)CC)=O)CC2(CNC(=O)C(F)OC(F)(F)F)CC1CCO2 33877,CC1CC(C(N2CC(C(N3CCC(N(C)C)C(C)C3)=O)C(C)C2)=O)CC(=O)N1 33878,c1(NC(c2ccc(CC)o2)c2nnnn2C(C)C)cncc(OCC(F)(F)F)c1 33879,C(c1ccc(OC)cn1)=CC(N1CCC(N(C(=O)CC2(C)CC2(Cl)Cl)CC)C1)=O 33880,CCCC(C(=O)N(CC(C)NC(C1(n2ccnc2)CCCC1)=O)C)C(C)C 33881,CCCC(C(=O)OC)C(=O)NC1CCC(CNC(=O)CC=CC(C)(C)C)CC1 33882,C1(NC(c2scc(C)c2)=O)CC(O)CN(C(=O)COc2ccc(C(N)=O)cc2)C1 33883,C1(N2C(NC(C(=O)N(CC)Cc3ccccc3)=O)CC2)CCCOC1 33884,N=c1nc(N2CCC(C3CC3)C2)[nH]c(=NCc2ccc3c(c2)CCCC3)[nH]1 33885,Cc1cc(C)c(C(=O)NC2CCN(C(c3ncccc3N)=O)C2C(C)C)c(=O)o1 33886,Cc1n[nH]c(=NCC(C)(C2CC2)NC(=O)C(C)Cc2ccccc2C)s1 33887,C(CC(F)F)(C(=O)N1CCC1C(=O)N(C)C)NC(c1cc(CCC)on1)=O 33888,C1(NC(c2c(SC3CC(NC(C)(C)C)C3)scc2)=O)CC2CCC1N2OC 33889,C1(NC(c2c(C)cnn2C)=O)CC2CCC1C(NC(=O)C(C)OC1CCCC1)C2 33890,C1(C(N(CCCNC(C2CSCN2C(C2CCCC2)=O)=O)C)=O)CC2CCC1O2 33891,CCC(F)(F)CC(=O)N1CC2(CNC(c3nccn3C(C)C)=O)CCC1C2 33892,CCC(CC(=O)N1CCC1COC)NC(=O)CCc1ccccc1O 33893,c1(CC)ncc(Cl)c(C(=O)NC2(CF)CCN(C(=O)CN3CC(C)(C)C3)C2)n1 33894,C1(O)(C(C)NC(Cc2c(C)con2)=O)CCN(C(c2cnc(N(C)C)o2)=O)C1 33895,CC1(C)OC2CC(C(=O)NC3CCOCC3NC(c3coc(Cl)c3)=O)CC2O1 33896,C1(C(N(CCN(C)C)Cc2c(F)cccc2Cl)=O)C2(CCC2)C12CCC2 33897,c1(C(=O)NC(CC)C(=O)OC)cc2n(n1)CCN(C(c1ccc(OC)nn1)=O)C2 33898,N1(C(c2c(OC)ccs2)C(=O)NCc2c(C)ncn2C)CC2CCCCC2C1C 33899,O=C1NCCc2cc(F)c(NC(C3CC(=C4CCC4)C3)=O)cc21 33900,c1(C(=O)NCC2(NC(=O)C=CC3CCC3)CC2)ccc2nc(S)oc2c1 33901,N1(c2nnc(N(C)CCO)s2)CCCC(C)(C(=O)NCCCN(C)C)C1 33902,N1(C(c2ccc(CCCCC)o2)=O)CC2C(C(=O)NC(C)C)C2C1 33903,C1(NC(c2cccc(C(C)=O)c2)=O)CC(O)CN(C(=O)C(n2nccc2C)C)C1 33904,C1(CC)CN(CCNc2ccc3c(c2)O3)C(C)CO1.c1(OC)ccccc1C 33905,Cc1nccc(C(=O)NCCCN(C)C(C2CNC(=O)N2C)=O)n1 33906,N1(C(COCCOC)=O)C(C(=O)N(CCCC(=O)OC)C)CCC12CC2 33907,C(=O)(CCCC(=O)N1CCOCC(CNC(=O)C(C)CC(F)F)C1)OCC 33908,C1(O)(C(N2CC(O)(CCNC(C3(C)CCC(C)C3)=O)C2)=O)CCCC(C)(C)C1 33909,CC(C)C(C)C(CNC(c1cnc[nH]1)=O)NC(C1CSC1)=O 33910,N1(C(C(CC)C)=O)CC(C)(CNC(C2(CC(F)(F)F)CC2)=O)CC1(C)C 33911,C(CC(N)=O)(C(=O)NCC1CCC2(CC1)CC2)NC(c1cccc(C)n1)=O 33912,Cc1cc(Cl)c(C(=O)N(C(C)(C)C2CC2)C(=O)Nc2cc(F)ccc2C)cc1F 33913,C#CCC(C)(C(=O)NC1(CCF)CC1)NC(C1CC2(CC2)CO1)=O 33914,c1(C(=O)NCC2(F)CC(NC(c3c(C)nc(CC)o3)=O)C2)cnc2sc(C)cn12 33915,c12ccc(cc1)oc2=O.C(=O)(C(C)=NOCC#N)N1C(c2c(C)ccs2)CCC1 33916,N1(C(C2=NOC(C)C2)=O)CCC2(CC1)CN(C(c1cn(C)cc1C(F)(F)F)=O)C2 33917,c1(NCCN(CC=C)C)[nH]c(=NC(COC)C(C)C)nc2c1ncn2C 33918,N1(C(=O)CCCc2nccs2)CCOC(Cc2ocnc2CC2CC2)C1 33919,c1(OCC)ccc(C(=O)NCC2(CNC(C3(C)CC3(C)C)=O)CCCC2)cn1 33920,c1(C(=O)NC(CC)CNC(C2CC3(CCC3)C2)=O)ccc(F)c(C)c1O 33921,CC(C)CC(C)CC(=O)NC(CNC(=O)Cn1cc(CN(C)C)nn1)CC(C)C 33922,c1(C(N2CCCC(CNC(C3(COC)CC(=C)C3)=O)C2)=O)cc(=N)[nH]c(Cl)n1 33923,C=CCC(CC(=O)NCCC1CC(OC)C1)NC(=O)C(N1CCNC1=O)C 33924,C(=O)(C#CC1CC1)N1C(C(=O)N(C2C(=O)NCC2)Cc2ccccc2)C(O)CC1 33925,N1(C(C2CCOC2c2ccccc2)C(=O)NC)Cc2ccccc2C(CO)C1 33926,N1(C(c2cc(C)c(C)o2)=O)CCN(C)CC1CNC(c1nocc1C1CC1)=O 33927,Cc1nc(C(N2CC(CNC(C3(C)CCCCNC3=O)=O)C2)=O)ccc1[N+](=O)[O-] 33928,C1(C(N2CCN(C)CC2)=O)CC(F)(F)CN1C(=O)CCc1cc(Br)ccc1F 33929,Cc1c(N(C)Cc2nnc(CO)s2)ncnc1N1C2CCCC1COC2 33930,C1(N(C(CC=C)=O)CCC)CCN(C(=O)C(C)C=C)C1 33931,N#CCCCC(=O)NC1C=CCC(C(N2CCN(c3ncccn3)CC2)=O)C1 33932,C1(OC(C)(C)C)CCC(OC(N(CCC(=O)NC)C(C)C)=O)CC1 33933,C1(CNC(=O)Cc2cccnc2)CC2(CO1)CN(C(=O)CCOC1COC1)C2 33934,CCC(CC(=O)N(C)CCNC(c1nccc(C)c1N)=O)C(F)F 33935,C(=O)(N=S(C)(=O)C1CC(O)C1)c1nc2n(c1)CC(C(=O)OC(C)(C)C)CC2 33936,C1(CN(C(=O)CC2(CO)CC2)C)COCCN1C(c1cc(-n2cccn2)ccn1)=O 33937,N1(C(CCCCC=C)=O)CC2(CCC2)CC1CNC(=O)C(C)C(C)C 33938,C1(OC)CC(CNC(=O)C(F)C(C)C)N(C(C2CC(F)C(=O)N2)=O)C1 33939,C1(NC(CNC(=O)CC2CCCC2)=O)CCCCN(C(c2ncsc2Br)=O)C1 33940,CC(C)C(C)(C)CNC(c1conc1C(C)NC(c1ncc(F)cn1)=O)=O 33941,Cc1cc(C(=O)NC2CCN(C(c3ccc(CN(C)C)[nH]3)=O)CC2)cc(F)c1C 33942,c1(OC)cccc2c1CC(C(N1CC(C)N(C(C)=O)CC1C)=O)CO2 33943,C#CCC(O)C(=O)NCCN(CC(C)O)C(C1CC(=C2CCC2)C1)=O 33944,C1(C(=O)NC(C(=O)OC)C(C)C)CC2CN(C(=O)Cc3ccc(O)nc3)CC2C1 33945,CC(CC(=O)NCCN(C)C(c1cnc2sccc2c1)=O)P(C)(C)=O 33946,N1(C(CC)=O)CCC(C2CCN(C(c3cc(F)c(Br)c(F)c3)=O)C2)CC1 33947,C(=O)(C(C)S(N)(=O)=O)N1CCC(NC(c2ccc(C)cc2)=O)C1C 33948,c1(-c2c(SC3(C(=O)OC)CCC3)ncnc2)ccccc1S(=O)(=O)NC 33949,C(C(C)CC(=O)N1CC2C(CNC(c3ccncc3SC(C)C)=O)C2C1)OC 33950,C1(CS(=O)(=O)NCC2CC(OCC(F)(F)F)C2)CC2C(C1)C2(F)F 33951,C(=O)(C1CCc2scnc21)N1CC(CN(C)C(c2ccn(C)c2)=O)C2(C1)CC2 33952,N1(C(COC)=O)CCc2nc(CNC(C3CCC4C(C3)C4(F)F)=O)sc2C1 33953,C1(NC(c2n(C)ncc2)=O)CC2CC1CN2C(c1ccncc1F)=O 33954,c1(C(=O)NCC2C(NC(c3c(N)cccc3F)=O)C2)ccc(F)cc1[N+](=O)[O-] 33955,c1(N2CCC(C(C)OC)CC2)cc(C)c(S(=O)(=O)NCC2CC2(Cl)Cl)cn1 33956,N1(C(COCC=C)=O)CC(NC(C2CCCCC(=O)N2)=O)CC12CCOCC2 33957,N1(C(c2cc(OCC)n[nH]2)=O)CCC2(CCCN(C(=O)CC3(CO)CC3)C2)C1 33958,C1(NC(Cc2cc(C)cc(C)c2)=O)CCN(C(=O)Cc2ccnn2C)CC(O)C1 33959,C1(O)(CNC(c2ccc(F)c(C3CC3)c2)=O)CCCN(C(c2cnn[nH]2)=O)C1 33960,c1(NC(N2C(C3(O)CN(C(=O)CC4CCCO4)C3)CCC2)=O)ccnc(Cl)c1 33961,C(=O)(C(CNC(c1cc(C)cc(C)n1)=O)CCC)NC(C#C)C1CC1 33962,c1(NCCC2(c3ccc(-c4cn(CCCC)nc4)cc3)CC2)c(C)cccc1F 33963,CC(C)CC(CC(C)C)C(=O)N(C)CC1CN(C(C2OCC2(C)C)=O)CC12CC2 33964,C1(NC(C=Cc2cc(OC)ns2)=O)CC2CCC(C1)N2C(=O)Cc1c[nH]nc1C 33965,c1(C(N2CCC(COC)(CNC(=O)C(F)CC3CC3)C2)=O)cn2c(n1)CCC2 33966,CC(C)CCC(C)N=c1[nH]c(=NC2COC3(CCC3)C2)c2sccc2[nH]1 33967,CP(C)(=O)C(O)C(=O)NCC1COCCN(C(=O)C(c2ccc(Cl)cc2)(F)F)C1 33968,N1(C(CNC(CCC2(O)CN(C(COCCC=C)=O)C2)=O)=O)CCCCCC1 33969,C1(NC(=O)CSc2nnnn2C2CCCC2)CCC(NC(C2(Cl)CC2)=O)CC1 33970,c1(CN(C)Cc2nn(CC)nc2C)ccc(C)cc1C 33971,C12(C(=O)NC(C3CCN(C(CCOCCOCC)=O)C3)(C)C)CCC(CC1)OC2 33972,c1(CC(C)C)ccc2cc(C(=O)NC3CCNCC3)[nH]c2c1 33973,c1(C(=O)NC2CCCCN(C(C3C(OC)CCCC3)=O)C2)cc2c([nH]1)CCOC2 33974,N1(C(C)C(=O)NCC2C3CN(C(C4CCC4)=O)CC23)C(=O)NC2(CCCC2)C1=O 33975,c1(C(=O)NC2CCN(C(c3c(OC)ccs3)=O)C2)ccc(C2CC2)c(OC)c1 33976,N1(C(C2(CC#C)CCCOC2)=O)CC2(CCN(C(=O)CC3CCCC3)CC2)C1 33977,C1(CNC(CN(C)S(N)(=O)=O)=O)CN(C(=O)Cc2ccsc2)CC1O 33978,C1(NC2CC(C)(C)OC2)CC1C1CN(C(=O)NCCS(C)(=O)=O)C1 33979,C(C(=O)NC1CC2(C1)CC2C(=O)NCC1(C#N)CC1)(C(C)C)NC(C)=O 33980,CC1CCC=C1C(=O)N1CCN(CCCNC(C2CC2Br)=O)CC1 33981,c1(CC(=O)NC2C3(CN(C(c4n(C)cnc4)=O)C3)CC2)cccc([N+](=O)[O-])c1 33982,Cc1csc(C(=O)NC2CN(C(=O)CCc3ccc[nH]3)CC2F)c1Cl 33983,c1(C(C)=O)cc(=NC2CCCC(NC(C3(C)CCCCCC3)=O)C2)[nH]c(Cl)n1 33984,N1(C(CCc2ccc(C)s2)=O)CCN(C(C2CCC=CCCC2)=O)CC1CO 33985,CC(C)(C)C(C)(O)C(=O)N1CCCN(C(c2coc(C(F)(F)F)n2)=O)C(CO)C1 33986,c1(C(=O)NC2CCCCC2NC(=O)C2=CCCS2)ccnc(Nc2ccccc2)n1 33987,C1(C(N(CC)Cc2ccc(O)cc2)=O)CCCN(C(c2cnoc2C)=O)CC1 33988,c1(C(N(CC(C)N(C(=O)Cn2ncc(O)nc2=O)C)C)=O)cc([N+](=O)[O-])nn1C 33989,C1(NC(c2c(C)n(C)nc2)=O)C(C)CN(C(=O)CC(C2CC2)C2CC2)CC1C 33990,C1(CNC(c2c(C)cc(O)nn2)=O)CN(C(c2ccc(F)cn2)=O)CCC1(F)F 33991,CC1(C)CN(Cc2ccccc2)CCC1NC(=O)NCCSCCCCN=[N+]=[N-] 33992,C1(CNC(c2c(C)scc2)=O)CC(NC(=O)CCc2cnn[nH]2)C1(C)C 33993,c1(OC)cc(NC(=O)C(C)N(C(C)(C)C)C(C)=O)c(Br)cc1Br 33994,C(c1cccc(F)c1F)=CC(=O)NC1CCCC(CNC(C(C)O)=O)C1 33995,CCC(C(C)C)C(C(=O)NCC)N1CCC(C(c2ccccc2Br)C)CC1 33996,C1(C(N(C)CCN(C(=O)C=CC(=O)NC2CC2)C)=O)CC(=O)N(C2CC2)C1 33997,C1(CC)CN(C(=O)C(F)OC(F)(F)F)CC1C(=O)N(C)Cc1ccc(F)cc1 33998,Cc1ccc2c(C(=O)N(C)CCN(C)C(C3SC4C=CC3CC4)=O)c[nH]c2c1 33999,N1(C(CNC(C)=O)=O)CCN(CCN(C)C(C2CC2Cl)=O)CC1 34000,C1(NC(N(C)C)=O)CC(CNC(c2coc(N(C)C)n2)=O)C12CCC2 34001,N1(C(Cc2cccc(C)c2)=O)CCN(C(=O)Cc2ccccc2F)CC(CO)C1 34002,C1(NC(CCOCCOC)=O)CCN(C(C2(c3ccc(C)nc3)CC2)=O)CC1F 34003,N1(C(C=Cc2cn(C)nc2)=O)Cc2ccccc2C1CNC(c1cnnn1C)=O 34004,c1(SC)nc(N2CCN(Cc3cccc(C)c3)CC2(C)C)c(Br)c(C)n1 34005,c1(OC)cccc(-n2cc(CNC(=O)CN3CC(C)(C)C3)nn2)c1C 34006,c1(OC)ccc(CC(=O)NC2CC(NC(c3csnn3)=O)C23CCC3)c(F)c1 34007,c1(C(=O)NCC2CC(F)CN2C(=O)C=CC2CCCC2)cc2cc(Cl)cnc2o1 34008,C1(C(=O)NC(COC)C)CC(O)CN1C(=O)CN1CCOCC1 34009,n1(CCOC)nc(CNc2ccccc2C)nc1-c1ccnc(OC)c1 34010,N1(C(CN(CCC)C)=O)CC2CCCC2(C(=O)NC2(CC3CC3)CCC2)C1 34011,C1(C(=O)NC2CN(C(C3(SC)CC3)=O)CC2O)CC(C)(C)OC1(C)C 34012,N1(S(=O)(=O)c2cccc(Br)c2)CCC2(CCCC2N2CCNCC(F)(F)C2)CC1 34013,C1(CN(C)C(c2[nH]nnc2C(F)F)=O)CCCN(C(C2(Cl)C(C(C)=O)C2)=O)C1 34014,N1(C(CC(C)C(F)F)=O)CC2(CCN(C(=O)C=Cc3ccn(C)c3)C2)C1 34015,C1(CCOC)(NC(c2ccon2)=O)CCN(C(C2CCOC2C)=O)C1 34016,C#CCCCC(C)C(=O)NC1CC(CNC(c2cc(F)c(N)cc2F)=O)C1 34017,N1(C(CN(CC)Cc2ccccc2)=O)CCCCC1CCNc1cnccn1 34018,C1(C(=O)OC)COC2(CCC2)CN1C(=O)CCCC1CCCC1 34019,N1(C(=O)Cc2ccc(Cl)s2)CC2CCCC(N=c3cnc(F)c[nH]3)C2C1 34020,N1(C(c2ncc(F)cc2F)=O)CC2CCN(C(C3CC4CCC3O4)=O)C2C1 34021,C12(CNC(c3ccc(Cl)cn3)=O)CC1CN(C(c1cccc(=O)o1)=O)C2 34022,N1(C(C2(OCC)CCC2)=O)CC(NC(c2cnc(C3CCCO3)s2)=O)C2(CC2)C1 34023,N1(C(CC2N(C(C(CSC)O)=O)CCC2)=O)CC2(CCCC2)C1 34024,c1(C(=O)NC2CC(NC(CCCC)=O)C23CCC3)cc2cnc(Cl)cc2s1 34025,c1(N(C)Cc2cccc(C(F)(F)F)n2)ccc(S(=O)(=O)NCC2(C)CCCS2)cn1 34026,c1(CCC)nc(=NCCCCC(C)NC(=O)C=C2CCCCCC2(F)F)s[nH]1 34027,c1(C(=O)NC2CCC(CNC(c3cc(C)oc3)=O)C2)ccc([N+](=O)[O-])n1C 34028,C12(NC(C(C)OCC=C)=O)CCCC1(F)CN(C(c1[nH]nc([N+](=O)[O-])c1Cl)=O)C2 34029,N1(C(C(C)c2cc[nH]n2)=O)CCC(C)C(CNC(=O)CSS(C)(=O)=O)C1 34030,c1(OC)cccc(C(N2CCC(N(C(=O)C=Cc3ccsc3)CCO)C2)=O)c1F 34031,C1(C(=O)NC2C(NC(CCC#C)=O)CCC2)CC2CCC(C1)C2F 34032,CC1CN(C(=O)CCCOC(C)(C)C)CCCN1C(=O)C(C)C#N 34033,C1(N(C)C)(C(=O)NCC(CNC(=O)C(F)=C2CCCC2)CO)CCCOC1 34034,C#CC1(NC(C2C=CC(NC(=O)CCCOCC)C2)=O)CCCCC1 34035,N1(C(C2(C)CCCCNC2=O)=O)CCOC2(CCN(C(=O)C=CC(N)=O)C2)C1 34036,C=CC(C)(O)CC(=O)NCC(C(=O)NCc1sc(C)cc1C)OC 34037,c1(OCCC)ccc(Cl)cc1CC(N1CC2C(NC(=O)C3=C(Cl)CC3)C2C1)=O 34038,c1(Oc2ccc(SC)c(Cl)c2)ccnc2cc(F)cnc12 34039,c1(OC)ccc(CNC(C(=O)NC(C)(C)C)C2CC2C)cc1C#N 34040,O=C1CCCC(C(=O)NC2COCCC2CC(=O)O)C1 34041,C1(C(=O)NC2CC(CNC(C3(F)CC4(CCC4)C3)=O)C2)CC2(C1)CC(F)(F)C2 34042,c1(C(N(CCOC)CCNC(=O)C(F)=CC2CC2)=O)ccc(C2CCC2(C)C)cc1 34043,C1(C(=O)NC2CCC(NC(c3ncc(C)cn3)=O)C2)Cc2ccc(Br)cc2C1 34044,C(=O)(C(C(=O)NCCCN(C)C(c1cncc([N+](=O)[O-])c1)=O)C(C)C)OCC 34045,N1(C(C2CCCCN(C(c3nc(CC)oc3)=O)C2)=O)CCC2(CCCCO2)C1 34046,C#Cc1ccc(CCC(=O)NC2CCN(C(c3cnn(C)c3)=O)C23CC3)cc1 34047,c1(C(=O)NCCNC(C(F)OC)=O)c(Cl)c([N+](=O)[O-])nn1C 34048,N1(C(C2CC23CCOC3)C(=O)NC(C)C)CCc2ccc(F)c(F)c2C1 34049,C1(C2CCN(C(C3C4(CC4)C34CC4)=O)CC2)(NC(c2ccn(C)n2)=O)CC1 34050,C1(NC(c2c(CC)onc2)=O)CCCN(C(c2coc(Cl)c2)=O)C1C 34051,CCC1=NOC(C(=O)NC2CC2NC(c2cn(CCF)nn2)=O)C1 34052,C1(NC(c2ncn(CC)n2)=O)CN(C(c2sccc2C(F)F)=O)CC1C 34053,CC(CN1CCOCC1)C(=O)NCCC1(O)CN(C(=O)Cc2cc[nH]c2)C1 34054,CCCCC(C(=O)N1CCSCC(C)C1)NC(C1CC2(CC(=O)C2)C1)=O 34055,c1(OC)ncnc(Cl)c1NC(=O)CC1(Nc2ccc(C)cc2Cl)CCC1 34056,C1(CNC(CCC(=C)C)=O)CN(C(C2CC2C(=O)OC(C)(C)C)=O)CCC12CCC2 34057,C1(CNC(c2cc(C)cc(O)n2)=O)CC2CCC(C1)N2C(=O)CC(O)CN(C)C 34058,Cc1ccc(Cl)c(C(=O)NC23CC2CN(C(c2ccc(C4CC4)nc2)=O)C3)c1 34059,CC1(C)OCCC1(O)C(=O)NC1CCC(C(=O)NC2(C3CCC3)CC2)CC1 34060,c1(C(N2CCC(N(C)C(c3csc(C(F)(F)F)c3)=O)C2)=O)cc(F)cc(F)c1 34061,N1(C(c2nc(C)oc2C)=O)CCCC2(C1)C(NC(=O)C(C)NC(N)=O)CCN2C 34062,c1(C(=O)NC2(C)CN(C(C=CCOC)=O)C2)ccc(S(=O)CC#N)cc1 34063,CC1(NC(C2CN(C(c3cc(N)cc(F)c3)=O)CCO2)=O)CN2CCC1CC2 34064,c1(CN(C(=O)C(CCc2ccccc2)C(=O)O)CC)cc(Cl)cc(Cl)c1 34065,C1(NC(C(C)OCCN(C)C)=O)CCSC12CN(C(=O)CCC1CCCO1)C2 34066,N1(C(C(=O)NCCNCC(C(F)(F)F)N2CCNCC2)=O)CC(C2CC2)(CO)C1 34067,c1(C(C)NC(c2c(C)n(C)cn2)=O)ccc2c(c1)CN(C(=O)C(F)C(C)C)C2 34068,Cc1c(C(N2CCCC2C2CN(C(=O)COCC3CCOCC3)C2)=O)cnn1C 34069,c1(OC)cnc(Br)cc1C(N1CC(F)CC1C(=O)NCCc1ccsc1)=O 34070,C1(NC(C2(CCO)CC2)=O)CCCN(C(C2(C(F)(F)F)CCOCC2)=O)CC1F 34071,N1(C(C(CC=C)C)=O)CCCC2(C1)CN(C(=O)CC1OCCOC1(C)C)CCO2 34072,C(N=c1ccc(-c2cccc(OC(F)(F)F)c2)c[nH]1)c1c(C)cc(Cl)cc1 34073,C1(NC(CN(C(=O)CN(CC(C)(C)C)C)C(C)C)=O)CCOC(C(C)C)C1 34074,c1(CC(=O)NCC2(CNC(CCOCCN(C)C)=O)CC2)nn(C)cc1Br 34075,Cc1nsc(C(=O)NCC2CCCN(C(=O)C(C)(C)C3CCC3)C2)c1N 34076,CCC(C)CCC(=O)NCc1ccc(C(N2CC(OCCF)C2)=O)s1 34077,CCC(CC(=O)Nc1cnn(CC2CC2)c1)NC(=O)CC1(C)CC1 34078,C1(CN(C(C(C)OCC)=O)C)CCCN(C(c2ccc(CC3CCC3)cc2)=O)C1 34079,N1(C(C(C)NS(CC)(=O)=O)=O)CC(NC(=O)CC2CC2)CC(C)C1 34080,C1(C(=O)NC(CN(C)C(=O)OC(C)(C)C)(C)C)CC(C2CC2)=NO1 34081,C=CC(C)(CC)OC.c12c[nH]nc1COC2=O 34082,N1(C(C2(NC(=O)OC(C)(C)C)CC=CC2)=O)CCCC(C2CCC2)C1 34083,N1(C(C(C)OCC)=O)CC2CCC(N(C)C(c3cnn4ccncc34)=O)C2C1 34084,C1(N(C(=O)C(=O)NC2CC2)C)CCC2CCN(C(c3ccccc3CO)=O)C1C2 34085,c1(OCC)cncc(C(=O)NCCC2CN(C(=O)Cc3cc(Cl)cs3)C2)c1 34086,C1(C)(CCNC(C2CCN(CC)C2)=O)CCN(C(c2ccoc2)=O)CC1 34087,C(=O)(CS(=O)(=O)C(C)C)N1C(CNC(C=CC=CCC)=O)(COC)CCC1 34088,c1(N2CC3(CN(C(c4c(OC)nccc4)=O)C3)C2)ncnc2scc(C)c12 34089,C1(CC(=O)NC(C2CC=CCC2)C(=O)N2CC(SC(F)F)C2)CCC=CCC1 34090,Nc1nc(C(=O)NC23CC(C2)N(C(=O)CCOCC(F)F)C3)ccc1O 34091,N1(CCC(=O)Nc2ccc(Cl)cc2)CCC2COCCC12 34092,CCC(C)(C)C(C)OC(C1CCCN1C(=O)OC(C)(C)C)=O 34093,C#CC1(NC(C2CC(NC(c3csc(F)c3)=O)C23CCC3)=O)CCCCC1 34094,N1(C(c2nc(COC)oc2)=O)C2CCC1CC(NC(=O)Cc1ccc(Br)cc1)C2 34095,C1(O)(CNC(c2cc(-c3ccc(Cl)cc3)no2)=O)CCN(Cc2ccsc2Br)C1 34096,C1(C#N)(C(=O)NC(C)C(CO)NC(c2cccnc2C(F)(F)F)=O)CC1(C)C 34097,Cc1csc(Cl)c1C(=O)NCCCN1CCN(C(=O)CSc2ccncc2)CC1 34098,c1(Cn2cc(CNc3cc(C)cc(C)c3)nn2)ccc2c(c1F)OCCO2 34099,Cc1c(C(=O)NCCC(C)(C)NC(C2CC2(C)C(F)F)=O)cnc2ncnn12 34100,n1(CC(=O)NCC(CNC(CC(CC)OC)=O)C)cccc([N+](=O)[O-])c1=O 34101,c1(C(C(C)C)SCC)nc(CC(C)(C)C)nn1-c1ccc(Br)nc1 34102,O=C(C(c1cccs1)=Cc1cccs1)NCC1CCC(CO)O1 34103,C1(CC(=O)N(C(COC)C)C)CCN(C(=O)CC=C(Cl)Cl)C1(C)C 34104,C(=O)(C1=CCCCCC1)N(C(CCCC=C)C)CCOC1CCC1 34105,c1(NC(N2CC(NC(C(F)=CC)=O)CC2(C)COC)=O)ccc2ccccc2c1 34106,N1(C(CC(C)=C(C)C)=O)CCC2CCCC12C(=O)NCCc1ccc(O)nc1 34107,C(=O)(C(C)(CNC(c1nn(C)cc1Cl)=O)CC)NCCOCC 34108,N1(C(C2ON=C(C)C2)=O)CCC2C(C1)CN2C(=O)CCCN1C(=O)CCC1=O 34109,c1(C(N2CC(C)N(C(C3CC(C(C)C)C3)=O)CC2)=O)cc2occc2n1C 34110,CC1C(NC(=O)C(C)(C)c2ncco2)CCCN1C(C1C(C)(C)C1(C)C)=O 34111,C1(C)(CC)C=C(C(=O)NC2CC(F)(CNC(c3cc(C)nc(O)n3)=O)C2)C1 34112,c1(C(=O)NCC2CCCN2C(C2CC(CF)C2)=O)cc2c(F)c(Cl)ccc2[nH]1 34113,c1(C(=O)NC(COC)CNC(c2cnnn2C2CC2)=O)cnc(Cl)n1C 34114,C(=O)(C1=CCCCC1C)N1CCCC(N(C(CCCOCC)=O)C)CC1 34115,N1(C(C2CCN(c3n(C)ccn3)C2)=O)CC2(CCN(C(C3CC3(C)C)=O)CC2)C1 34116,C(=O)(CCCS(=O)(=O)NC(c1nc(C)no1)C1CC1)OC 34117,O=C(C1CCCc2ncnn21)NCC1CCN(C(c2ccnn2C2CCC2)=O)C1 34118,C1(CNC(C(C2CN(C(c3cc(OCC)n[nH]3)=O)C2)OC)=O)CCCCN1C 34119,C1(F)(C(=O)OC)CCN(C(=O)COC)C1.c12ccc(cc1)OC(=O)N2 34120,N1(C(C2CC(C)CN2Cc2ncccc2O)=O)CC(CO)C2(CCC2)C1 34121,c1(OC)c(C(=O)NCC2(NC(C3CC=CCC3)=O)CCOC2)ccc(Cl)c1Cl 34122,C1(NC(=O)NCc2ccc(S(C)=O)cc2)CCC(F)(F)C(C)(C)O1 34123,c1(C(=O)NCC(CCOC)NC(C2CC3CC3C2)=O)oc(COC)nc1C 34124,CC1CCCCN1CCC(=O)NCC1CC1NC(c1ccc(SC(F)F)cc1)=O 34125,C(=O)(C(CC(C)C)N(C)C)NC1(CC(N2CCCC(CCC#C)C2)=O)CCC1 34126,C(=O)(C1=C(SC)CCCC1)NCC(C1CCC1)NC(C(CC)CCOC)=O 34127,N1(C(c2ccc(-c3cnn(C)c3)s2)C(=O)NCC)CC(CSC)C1(C)C 34128,c1(C(=O)NC23CC2CN(C(c2cnc4sccn24)=O)C3)c(F)ccc2n[nH]cc12 34129,N1(C(C(C)NC(CC)=O)=O)CC(N(C)C(c2n[nH]c(C)c2O)=O)C(C)(C)C1 34130,c1(CC(=O)NCCNC(C2CCSCC2)=O)noc2ccc(Br)cc12 34131,N1(C(C2N(C)CCN(C(C(c3ccn(C)c3)C)=O)C2)=O)CCCC(C)(C)CC1 34132,C1(CC(C)(C)C#N)C(=O)N1.N1(CCS(C)=O)CCC(SC(F)(F)F)CC1 34133,Cc1c(C(=O)N(C2CN(C(=O)COCC3CCC3)CC2O)C)oc2ccccc12 34134,c1(-c2ccc(CC)o2)nc(C2CCC2)nn1CCCO 34135,C1(C(=O)Nc2c(C)cccc2CO)CCN(C(=O)COCC2CC2)C12CCC2 34136,c1(NC(C2C(NC(c3cc(-c4ccco4)on3)=O)CCC2)=O)ccc(Cl)cc1Br 34137,C1(C(N2CCCC(Cn3cc(C(CC)O)nn3)C2)=O)CCc2nc(O)[nH]c2C1 34138,c1(NC(C)=O)ccc(NC(c2nnnn2CCC2CC2)C2CC=CC2)cc1 34139,CC(C)C(C)C(C)CC(=O)NC(C)CC1CCN(C(=O)Cn2cnc(=N)[nH]2)CC1 34140,CCCC(O)C(=O)NCC(C1CCN(C(C2(C)CCNC2=O)=O)CC1)O 34141,N1(C(CCC(N)=O)=O)CC(CNC(=O)CC(O)Cc2ccccc2)C2(CCC2)C1 34142,C1(NC(C(COCC)(C)C)=O)COC2CN(C(=O)C(F)C(C)(F)F)CC12 34143,C(=O)(C1CC(=O)c2ccccc21)N1C(C)(CNC(C(C)NC(N)=O)=O)CCC1 34144,Cc1cc(C(=O)N(C2CN(C(C3(C)CCCCCC3)=O)CC2(C)C)C)nc(C)c1 34145,C=CC(C)(CC)C(=O)N(CCCNC(=O)CNC(=O)COc1ccc(F)cc1)C 34146,Cc1cncc(C(=O)NC2CCCC2NC(=O)CCF)c1Cl 34147,c1(C(=O)NC(C)(CNC(=O)CC2CC=CCC2)CO)cc(Cl)ccc1O 34148,C1(NC(c2c(C)onc2)=O)CN(C(=O)CN2CSCCSC2)CC(C)(C)C1 34149,Cc1oc(Cl)nc1C(=O)NC1(CCCC(=O)NC2CC(C(F)F)C2)CCC1 34150,CC1CC(NC(=O)C(C)S(N)(=O)=O)CN(C(=O)C(C)(C)F)C1 34151,N1(C(=O)Cc2c[nH]nc2O)CCC2CCN(C(c3ccc(Cl)cc3O)=O)CC2C1 34152,N1(C(c2c(C)[nH]cc2)=O)CC(NC(C2CCC(N(C)C)CC2)=O)C2CC12 34153,C1(NC(C2CCC3CC23)=O)CN(C(c2cnc(Br)s2)=O)CC12CC2 34154,C1(NC(=O)COC2CCOC2)CC(F)CN(C(c2c[nH]nc2C(F)(F)F)=O)C1 34155,C1(NC(CN2CCC(C)(C)C2)=O)CN(C(C2(C)CC3CC3C2)=O)CC12CC2 34156,C(=O)(CCC(=O)NCC1(CNC(C2CC2C(F)F)=O)CC1)c1cn(C(C)C)nc1 34157,CC(C)CC(C)(O)C(=O)NC1CC(CCNC(=O)Cc2ccn(C(C)C)n2)C1 34158,C(=O)(C(C)(C)Cc1cnn[nH]1)N1CC(CNC(c2cc(COC)[nH]n2)=O)(OC)C1 34159,c1(CNC(C2(C)CCN(C(c3cc(C(C)=O)cn3C)=O)C2)=O)ccn(C)c(=O)c1 34160,CC1=CC(O)CN(C(=O)NC(c2nc(C(C)CC#N)cs2)=O)C1 34161,C1(CNC(=O)CN2CCOCC2)CC(F)(F)CN1Cc1ncc(Cl)cn1 34162,c1(C(=O)NC2CN(C3CCCN(CC)C3=O)C2)cc2ccc(Cl)cn2n1 34163,c1(SC)ncc(C(=O)NC(CO)C(C)NC(c2ccncc2C)=O)c(O)n1 34164,Cc1cc(Br)ccc1CN1CC(CO)(NC(c2ncc(Cl)nc2Br)=O)C1 34165,C1(NC(C2(CCC)CC2)=O)CCCC1NC(=O)C(C)(C)C1CCCCO1 34166,C(=O)(C(F)C(C)(F)F)NC1C(CNC(C2(CC#C)CC=CCC2)=O)CC1 34167,c1(OC)cc(C2CCN(C(C3(C)CCN(C(C)=O)C3)=O)CC2)cnc1OC 34168,C1(C(C)C)CCC(C(=O)N(CCNC(=O)C(C)N2CCC2)CCN(C)C)CC1 34169,c1(CC)noc(C(=O)NC2CCN(C(C3CC(OC)C3)=O)CC2)c1C 34170,c1(C(N2C(C)(C)C(CNC(C3CC(=O)N3)=O)CC2)=O)cnc2c(c1)NCC(=O)N2 34171,c1(C(C(=O)NCCC)N(C)C(c2cccc(OC)c2)C)cn(C2CC2)nc1C 34172,CCC(O)C(C)(C)C(=O)N1CCN(C(=O)C(C)(Cl)Cl)CC(O)C1 34173,c1(C(=O)NC2C(C(=O)NC(CC=C)C(=O)OCC)CC2)cc(C)nc(O)n1 34174,c1(CNCc2cccc(C(=O)OCc3ccccc3)c2)cc(CCO)cc(Br)c1 34175,Cc1ccsc1CC(N1CCC1(C)CC(=O)NCCC1CC1C)=O 34176,C1(SCC)CC2(CC(=O)CC(C)(C)O2)O1.C(CCOCCN(C)CC)O 34177,N1(C(C(C=C)(C)CC)=O)CCCCC12CN(C(c1ccc(C(=O)OC)s1)=O)C2 34178,O=C(C1Cc2ccccc21)N1CCC(N2CCN(C(C3(CO)COC3)=O)CC2)C1 34179,N#CC1(C(=O)NC2CC(NC(C34CCOCC3C4)=O)C2)CCSCC1 34180,N1(C(=O)COC2CC2(F)F)CCC(NC(=O)COCc2c[nH]nc2C(F)F)CC1 34181,N1(C(C(CSC)OC)=O)CC(O)CC1C(=O)NC1CC=CCC1C 34182,c1(C(N2CCC(Cn3cccc3)CC2)C(=O)NCC=C)nn(C(C)C)nc1Br 34183,Cc1cc(Br)cc(C(=O)NC2(CCO)CN(C(C3CC(C)CO3)=O)C2)c1C 34184,N1(C(CC(C)(C)N(C(c2cc(SC)oc2)=O)C)=O)CCCCC(C)C1 34185,C1(C)(C(N2CC(NC(c3c(C)occ3C(F)(F)F)=O)C2)=O)OC(C)(C)OC1C 34186,C(=O)(C1CSc2ccccc21)NCCC1(C)CCN(C(C2CC(O)C2)=O)C1 34187,C1(CNC(CCCC#CC)=O)CC12CCN(C(C1CC3CCC(C1)N3C)=O)CC2 34188,C1(C(=O)NCC(COC)NC(CC2N(CC)CCC2)=O)CCc2cnnn2C1 34189,N1(C(C(COC)C(F)(F)F)=O)CCCC2(NC(=O)CS(C)(=O)=O)CCCC12 34190,N1(C(c2cnc(C3CCC3)o2)=O)CCN(C(c2cnn3c2OCC3)=O)C(CO)C1 34191,c1(CC)ncc(C(=O)NC2CC3CN(C(c4ocnc4C(F)F)=O)CC23)c(O)n1 34192,CC1(C)CCCC(C(N2CC3(CC(CNC(=O)Cc4cn[nH]c4)C3)C2)=O)C1 34193,C(C(=O)NCC1CC(C)N(C(c2ccccc2SCC#N)=O)C1)(C(C)C)OCC 34194,c1(C(=O)NCC(=CC(=O)NC(CC=C)CO)C)n[nH]c(C)c1Cl 34195,C1(NC(c2coc(C(F)F)c2)=O)(CF)CCN(C(c2cncnc2)=O)C1 34196,C(C1=NOC2COCC12)NC(=O)NC1CC(=O)N(C2CCCCCC2)C1 34197,C1(CCNC(C(C)(C)OC)=O)CN(C(=O)C(C)NC(c2ccoc2)=O)CC1C 34198,N1(C(C2C(C)OCCO2)=O)CCCC(C)(C(N2CCC2CC2CC2)=O)C1 34199,CC1CC(NC(=O)CC(C)(C)F)CN(C(c2cncnc2)=O)C1 34200,c1(C(N(CCNC(C2(C)C(C)CCC2)=O)CC2CC2)=O)cnn2c1CCC2 34201,c1(NC(C2CC3CC3N2C(=O)CCN2CCOCC2)=O)cccc(C(F)(F)F)c1 34202,N1(C(CC=C=C)=O)CC2CC1C2NC(c1ccccc1)=O 34203,N1(C(c2n(CCOC)ncc2)=O)CCCC1(C)C(C)(C)CNC(=O)C(F)C1CCC1 34204,c1(C(=O)NC(COC(C)C)C(=O)NC2C=CCCCC2)nnn(C)c1N 34205,C1(C(F)(F)F)(OC)CCCN(C(C(=O)NC(C)C)c2nccs2)C1 34206,c1(OC)ncccc1-c1cn(CCCNC(=O)C(C)(C2CC2)OC(=O)C2CC2)nn1 34207,C1(C(=O)NC2CC(NC(c3c(C)nsc3)=O)C2)C2CN(C(=O)OC(C)(C)C)CC12 34208,CCC(CCOC)C(=O)N1CCC(CN(C)C(C2COC(=O)N2C)=O)C1 34209,C(=O)(C(C)(C)CC(F)(F)F)NCCCC(CCC)Nc1ncc(O)cn1 34210,N1(C(C(c2ccccn2)C)=O)CCN(C(c2ccc(Cl)cc2N)=O)CC1C 34211,c1(C(=O)NCC2N(C(c3c(CC)nns3)=O)CC(O)C2)cnc(C)cc1Cl 34212,C1(C(=O)NC)COCCN1C(c1cc(C2CNCCO2)no1)=O 34213,c1(C(=O)NC(C2(O)CCN(C(CSc3cc(C)on3)=O)C2)C)cccc(=S)n1O 34214,c1(C(=O)NC2(CC(=O)Nc3ccc(C)cn3)CCC2)cc(F)c(F)cc1C 34215,c1(C(=O)NC(C2(O)CN(C(C(CC)N(C)C)=O)C2)C)cc2nccnc2cc1C 34216,C=Cc1cncc(C(=O)NC(C2CCOC2)CNC(c2c(C)cnnc2O)=O)c1 34217,N1(C(C2CC(n3ncc(OC)c3)C2)=O)CCC2(COC(C)C2)C1 34218,c1(C(=O)NCC2CCN(C(CN(C(COC)=O)C)=O)CC2)ccc(Cl)cc1Cl 34219,C1(NC(C2CCC=CO2)=O)CN(C(=O)COc2ccon2)CC12CCOCC2 34220,c1(OC)c(F)ccc(F)c1C(=O)NC1CC1CNC(=O)CC1CCC2(CCC2)O1 34221,C1(C(=O)NCC2(C)CC(F)(F)CN2)CCc2n[nH]cc2C1 34222,c1(CN2CC(C)CC(NC(CC=CCC)=O)C2)coc2ccccc12 34223,C(=O)(C(F)(CNC(C1(C#N)CCCOC1)=O)C(C)C)NC(C(=O)N(CC)CC)C 34224,N1(C(c2c(C)con2)=O)CC(NC(c2cccc3cnsc23)=O)C2(CCC2)C1 34225,C(C(CC(C)C)C(=O)Nc1cnc(C)c(C#N)c1)NC(C1(OC)CCC(C)C1)=O 34226,N1(c2nc(Cl)nc(C)c2F)CCC2(CC1)OCCC2NC(=O)Cn1nnnc1C 34227,c1(CN2CC(OC)C(NC(=O)CCOCC3CC3)CC2)ccc2nc[nH]c2c1 34228,C1(CNC(c2scnc2Cl)=O)CCCC1NC(=O)C(Cc1ccccc1)C1CC1 34229,N1(C(CC2CC(=C)C2)=O)CCN2CCOCC2(CNC(=O)C(C)CCCOC)C1 34230,c1(CNC(COCC#C)=O)c[nH]nc1NC(=O)C1CC1.C12(CC1)CS2 34231,CC(C)CCC(F)C(=O)NC(C)(CNC(c1cccc2nccn12)=O)CO 34232,Cc1cc(C(N2CCCC(N(C(=O)C(C)CC3CC3)C)C2)=O)ncc1Cl 34233,CC1OC(=O)NC1C(=O)NC1CCCC(NC(c2cc(Br)sn2)=O)C1 34234,c1(SC)cc(NC2CCN(C(=O)C(C(C)C)n3cnnc3)CC2C)nc(SC)n1 34235,N1(C(C2CCC(=C)CC2)=O)CCC2CCN(C(c3cc4sc(Cl)cc4[nH]3)=O)CC12 34236,Cc1noc(C)c1C(C)C(=O)NCCC(C)NC(=O)C(C)C1CCCO1 34237,c1(NC(C2C(N(C(=O)C=CCN3CCCCC3)CCN)C2)=O)cnncc1Cl 34238,N1(C(C2N(C(CC3C(C)C(=O)CC3)=O)CCCC2(C)C)=O)CC23CCC2(COC3)C1 34239,c1(C(N(C(C)CNC(=O)C(c2cncnc2)C)C)=O)cnc2cnn(C)c2c1 34240,CC(N=c1cc[nH]cc1S(=O)(=O)N1CCCC(CN(C)C)C1)c1ccc(Br)o1 34241,Cc1ccc2nc(C(=O)NC3COCCN(C(C4CCCSS4)=O)C3)cn2c1 34242,C(=O)(CC(C)C1CC1)NCC1C(NC(COCC(C)C)=O)C1 34243,C1(O)(C(NOC)=O)CCCN(CC(C)OC)CC1 34244,N1(C(Cc2c(C)noc2)=O)CCC2C1CCCN2C(C1CCCCO1)=O 34245,C(CC(O)C(=O)NC1(c2ccccc2)CN(C(c2cc(C)on2)=O)C1)SC 34246,c1(C(C(=O)NCCC(=O)OCC)N(c2ccccc2)C)nc(Cl)sc1Cl 34247,C=CC(CC)C(=O)NCCC1(C(=O)N(C)CC2CC2C)CCC1 34248,C(CC(C(=O)NC(CCO)c1ccco1)NC(C1CN(C(C)=O)C1)=O)SC 34249,S(=O)(=O)(c1ccc2c(c1)CCN2CC)N1C(C(=O)NC(CCCC)CO)CCC1 34250,c1(SC)cccc(-c2cncc(CNCc3ncccc3Br)c2)c1 34251,c1(C(=O)NCC2N(C(C=NOC)=O)CCC2)cccc(C#N)c1 34252,N1(C(C(C)O)=O)CCC(C2CC(NC(=O)CCc3ccn(C)n3)C2)CC1 34253,C1(CNC(C2CC(C#C)(O)C2)=O)CC(C(=O)N2CCCN(C(N)=O)CC2)=NO1 34254,N1(C(c2c(C)nc(C)o2)=O)CC2CCN(C(=O)CC3CCCNC3=O)CC12 34255,c1(C(=O)NCCN(C(c2c(C)ccc(C)c2)=O)C)nc2ccccc2cc1CO 34256,C(=O)(C(C)(C)S(C)(=O)=O)N1CC(CCNC(c2c(OCC#N)cccc2)=O)C1 34257,C(=O)(C1=CCCC1(C)C)N1CCN(C(Cn2cc(C(C)=O)nn2)=O)CC1CO 34258,C1(NC(C2(CC)CCOC2)=O)CCCCCC1NC(=O)C(F)(F)c1csc(C)c1 34259,Cc1ccccc1C1(C(=O)NCC(C)CNC(C2(C)CSC2)=O)CC1 34260,N1(C(COCCCC#C)=O)CCC(F)(F)C(CNC(c2sccc2COC)=O)C1 34261,C(N=c1cc2n([nH]1)CCCC2)(c1c(CCc2[nH]ccc2)ocn1)c1nn[nH]n1 34262,C(=O)(C(C#N)C(C)C)N1CCCC(NC(Cc2c(C)cnn2C)=O)C1 34263,C1(CC)CN(C(C2(CO)CCCC2)=O)CCN1C(c1csc(-c2cccs2)n1)=O 34264,c1(C(N(CC(CC)NC(C(CC=C)NC(C)=O)=O)CC)=O)cc(F)ccc1C 34265,N1(C(CCN(CCC)C)=O)CC=C(C(C)(C)C(=O)NC2CC(C3CC3)C2)C1 34266,C=CCC(CNC(=O)C(C)N(C1(CC(=O)NC)CCC1)CC)NCC(=O)NCC 34267,C1(OC)(CNC(c2cnoc2C)=O)CCN(C(=O)C2=COCCC2)CC1 34268,N1(C(c2c(SCC)cncc2)=O)C2CCC1C(CNC(=O)Cn1ccnc1C)C2 34269,N1(C(C2(NC(=O)CC3C=CCC3)CCSC2)=O)CCC12CCSCC2 34270,c1(CC(=O)N(CC(C)C)CCN(c2ccccc2)C)ccccc1-c1nn[nH]n1 34271,C1(CNC(C=CC2N(C)CCC2)=O)CN(C)CCN1Cc1ccccc1 34272,C=CC1CN(C(=O)COCC(F)F)CC1NC(=O)CCc1ncc(F)cn1 34273,c1(C(=O)NCCCNC(C2CC(P(C)(C)=O)C2)=O)n[nH]c2ccc([N+](=O)[O-])cc12 34274,N1(C(c2c(CC)cccc2)C(=O)NCCOC)CC2(C)CC1CCO2 34275,N1(C(C2CCN(Cc3c(OC)ccc(Br)c3)CC2O)=O)CCC2(CC1)CN(C)C2 34276,NS(=O)(=O)c1ccc(CC(=O)NC2CCC2NC(C2(CC3CC3)CCC2)=O)cc1 34277,C1(NC(CC2CC(OCC)C2)=O)CC2(CC2)CN1C(=O)CNC(=O)CCC(C)C 34278,Cc1nccc(C(N2CCC(NC(c3cc(Cl)cnc3O)=O)C(C)C2)=O)c1C 34279,C1(C(=O)NCCC(C)N(C)C(c2cn(C)nn2)=O)CCC(C)(C)C1 34280,C1(NC(Cn2nc(C)n(C)c2=O)=O)CC12CCN(C(C1OCCC1(C)C)=O)CC2 34281,N1(C(c2cc(C)oc2C(F)(F)F)=O)CCN(C(c2cnc(O)o2)=O)CC(C)(F)C1 34282,Cc1cc(NC(=O)NC2(c3ccccc3)CCOC2)cnc1C 34283,CCC(C(=O)NCC1(C)CCCN1C(=O)C1=NOC(C(C)(C)C)C1)C(C)C 34284,c1(CCC(=O)NC(C2CCN(C(c3c(C)nn(C)c3)=O)C2)C)c(Cl)cccc1Cl 34285,CCCN=C(NCc1ccc(C(=O)OC(C)(C)C)c(Cl)c1)NCC.C12CCN1C2 34286,C1(C(=O)NCCC2(C)CCN(C(C3C4C5CCC(C5)C34)=O)C2)C2CCC3C(C2)CC13 34287,C1(NC(C(n2c(C)ncc2)C)=O)CN(C(=O)Cc2cncs2)CC12CCC2 34288,C(=O)(C1=C(C)OCCS1(=O)=O)NC1CN(C(C(CC)CC(F)F)=O)CC1C 34289,c1(C(=O)NC2CN(C(C(C)N(C)C)=O)CC2C)cc(F)c2nc(O)ccc2c1 34290,C1(CC)CCC(C(N2CCCC(CNC(c3nnn(C(C)(C)C)n3)=O)C2)=O)CC1 34291,C1(NC(c2c(C(C)C)scn2)=O)CN(C(c2c[nH]ccc2=O)=O)CC2(CCC2)C1 34292,C(C(C)C(=O)NC(C(=O)NC(C1CCOC1)CO)C1CCCC1)OC 34293,C1(C(N(c2ccccc2)CC)=O)CC12CCN(C(=O)CC1CCCC(=O)C1)CC2 34294,Cc1cc(Br)ccc1CC(=O)NC1CCC1NC(C1CCCCN1C)=O 34295,c1(SC2(CN)CCOCC2)ncc(Br)cc1OC(CC)C(=O)NC1CCOC1 34296,C1(C(=O)NCCCCC2CN(C(c3c(C)cc(C)[nH]3)=O)C2)CC12CCCOC2 34297,c1(OC)cc(C(=O)NC2CCN(C(c3cc(C)c(C)[nH]3)=O)C2)c(N)c(Br)c1 34298,C=CCC(C(=O)N1CC(C(=O)N(CCCN(C)C)CC)CC(C)C1)C(C)C 34299,C1(NC(C=C(CC)CC)=O)CCCC1NC(=O)CC1(CO)CC1 34300,Cc1nc2cc(C(N3CCCC(F)(F)CC3)=O)ccc2n1C(C)CO 34301,C1(C(N(CC(=O)NCC)C)=O)CCCN(C(=O)COC2CC2)CC1 34302,N1(C(CCC(=O)OCC)=O)CCC2(CCCN2C(=O)Cn2cc(C)cn2)C1 34303,CCCC(C(=O)NCCCOCCNC(C1CCc2nncn2C1)=O)S(N)(=O)=O 34304,N1(C(C(F)=CCC)=O)CCCC(NC(=O)COCC2CCCO2)C1C 34305,N1(C(c2nc(Cl)cs2)=O)CC(C2(N=c3[nH]nc(C4CC4)o3)CC2)C1 34306,C1(C(=O)NCC(C)CN(C)C(c2ncsc2C2CC2)=O)COC2(CCC2)C1 34307,C(=O)(C(CNC(=O)Cn1cccc1)CC(C)C)NC1CC(OC)C1(C)C 34308,N1(C(c2c(C)nns2)C(=O)NC(C)(C)C)CCCC(F)(CO)C1 34309,N1(C(C(C)(C)O)=O)CC2OCCN(C(c3c[nH]c4nccc(Br)c34)=O)C2C1 34310,C1(C(F)(F)F)(C(=O)NC(CCNC(Cc2c(C)scc2)=O)C)CC2CCC1C2 34311,CC(C)C(O)C(=O)NCc1ccc(C(=O)N(C)CC2(F)CCC2)o1 34312,N1(C(CC2(C)N(C(c3cnc(CC)o3)=O)CC2)=O)CC(=O)NC(C)C1 34313,c1(C(=O)NCC(CC)NC(c2cc(F)cs2)=O)ccnn1C(F)F 34314,N1(C(C(C(C)(C)C)OC)=O)CCCC(C2CN(C(=O)C(=O)NCC3CC3)C2)C1 34315,N1(C(c2c(CC)nn(C)c2)=O)CC2CC1CN(C(c1nocc1Cl)=O)C2 34316,Nc1cc(Cl)cc(Cl)c1C(N1CCC(NC(=O)CCc2cncc(F)c2)C1)=O 34317,C(CC(C)C(=O)NC(C)CC1CN(C(=O)CCc2conc2C)C1)=CC 34318,CC1CN(C(C2CCCN2C=O)=O)CC1NC(C1(N(C)C)CCC1)=O 34319,CC1OCCC1(C)C(N1CCC(C(=O)NCC(C2CC(C)(C)C2)O)CC1)=O 34320,C1(NCc2nnc(-n3ccnc3)o2)CCN(C2CCCCC2)C1=O 34321,C1(CN(C)C(C2(S(N)(=O)=O)CC2)=O)CC(F)CN1C(=O)CSc1n[nH]c(O)n1 34322,c1(SCC)ccccc1CC(=O)NCC1(C)CCCC1NC(=O)C(C)OC 34323,c1(C(N(CC(C)NC(C(CNC(C)=O)(C)C)=O)C)=O)cc2sccc2cn1 34324,c1(NCC2CC(C)SCC2)[nH]c(=NCc2cc(C3CC3)ccn2)nc2sccc12 34325,c1(C(N(C(c2ccccc2)CNC(c2onc(C)n2)=O)C)=O)ccc(O)nn1 34326,c1(C(=O)NC2C(CNC(C(CC)CC3CCCC3)=O)CC2)ncc2ccccn12 34327,C(N=c1ccnc(C2CC2)[nH]1)c1c(CN2CCN(S(C)(=O)=O)CC2)cncc1 34328,c1(CN(C(C2CCCN(C(c3coc(C)n3)=O)C2)=O)CC)ccc(O)cc1 34329,N1(CCSc2ccc(C(C)C)cc2)CCCN(C(=O)C(C)C#N)CC1 34330,c1(OC)cc(C(=O)NCCC(C)(C)C#N)sc1Cl 34331,N1(C(CC(C)(C)O)=O)CC2(CC(C(=O)Nc3ccc(F)c(F)c3)CO2)C1 34332,c1(CC(=O)NC(C)(C)CCNC(c2cc(C(N)=O)[nH]n2)=O)cccc(F)c1O 34333,C(=O)(CC(C)CC(F)(F)F)N1CC(C)C(NC(c2cc3cc(Cl)ccn3n2)=O)C1 34334,C1(CNC(C(CC)C)=O)CCCCN1C(c1cccc(-c2ccoc2)c1)=O 34335,N1(C(c2c(C)cccn2)=O)CC(C)CN(C(c2ccc(F)c(N)c2F)=O)C(C)C1 34336,N1(C(c2ccccc2)C)CCCC(C)(C(=O)NCCNC2(C(F)(F)F)CC=CC2)C1 34337,c1(CC(=O)NC2CCC(NC(C3C(C)(C)C3)=O)CC2)ccc(S(N)(=O)=O)cc1 34338,c1(C(N(CC(=O)NC)C)=O)ccc2c(c1)CN(C(c1ccc(C)cc1)=O)CC2 34339,C1(NC(COCCC)=O)CN(C(=O)CCc2scnc2C)CCC1F 34340,C1(CNC(CCC(=O)c2ccc(C)s2)=O)CN(C(=O)C(C)(C)CC#N)CCC1C 34341,C(C(CC(=O)NCC1(CF)CC1)NC(=O)C(C)(C)CSC)OC 34342,C(=O)(CCCCc1ccccc1OC)NC(CC)(C)C#N 34343,N1(C(C(C)(C)OCC)=O)CCCC(C)(C(=O)NC(C)CCC=C(C)C)C1 34344,c1(CC(=O)N(C2CCCN(C(c3cccnc3)=O)CC2)CC)c(F)cncc1Cl 34345,C1(C(=O)NCCCCNC(CN(CC(=O)NC(C)C)C)=O)CCc2nc(C)cn2C1 34346,C(=O)(C(C(CC)CC)OC)N1CC(N(C(=O)C(c2cnn(CC)c2C)=O)CC)C1 34347,c1(C(=O)NC2C(NC(C=CCOC)=O)C2)cccc2oc(C)cc12 34348,c1(C(=O)NC2CCC(N(C(c3c(C)ocn3)=O)C)C2)cnc2c(c1)CCOC2 34349,C1(NC(C(C)N(C(C2COCCC2C)=O)C2CC2)=O)CC(C2CCCC2)C1 34350,C1(c2ccc(Br)cc2)(NC(c2c(CC)nc(C)s2)=O)CCC(C)(C)C1 34351,C1(COC)(NC(=O)CCC=C(C)C)CCN(C(=O)C(c2ccccc2)SC)C1 34352,c1(C(=O)NC(C(C)(C)OC)C)ccc(CNC(=O)Cn2cc(C#N)cn2)nc1 34353,c1(C(=O)NC(CSCC)CO)cnc(CNC(c2ccnn2C(C)C)=O)nc1 34354,N1(C(C(C2SC(=N)NC2=O)C)=O)CC2OCCN(C(C3CN(C)CCO3)=O)C2C1 34355,C(c1cccc(C)c1)=CC(N1CCCC(CN(C(=O)C2=CCCC2C)CC)C1)=O 34356,N1(C(c2cc(C(C)C)no2)=O)CCN(C(=O)CCCNS(C)(=O)=O)CC2(CC2)C1 34357,C1(NC(c2cc(CC)ncc2)=O)CCN(C(=O)Cc2cncnc2)CC(C)(C)C1 34358,N1(C(C(Br)=C(C)C)=O)CC(CNC(C2CNC(=O)C2)=O)C(F)(F)C1 34359,c1(COC)nn(C)cc1C(=O)Nc1cccc(-c2nc(C)co2)c1 34360,N1(C(c2nc(CCC)oc2)=O)CCC(CC)C1CNC(C1CC(F)C1)=O 34361,N1(C(N2CC(C(=O)NCC3CCOC3CC)C2)=O)CCCOC(C2CC2)C1.C1CC1 34362,N1(C(C(C=C)c2ccccc2)=O)CCN(C(c2cnc(CC)s2)=O)CC1CC1CC1 34363,n1(CC)nc2c(c1C(=O)NC(C)CCN(C)C(C1CC1CC(C)C)=O)CCCC2 34364,c1(OC(C)C(=O)NC2COC2)cccc(CO)c1F 34365,CCCCC(C)(F)C(=O)NCC(C)N(C(=O)CN1CCOCC1)C 34366,N1(C(CCN(C)CC)=O)CCC2C(NC(c3nn(CC)cc3Cl)=O)C2CC1 34367,N1(C(C(CC)N(CC)CC)=O)CC2CCC(CNC(=O)C=CSC)CC2C1 34368,C1(NC(c2ccc(SC(C)C)cc2)=O)CC2CC1CN2C(=O)CN(C)CCO 34369,c1(C(=O)NCC(CN(C(CNC(=O)NC)=O)C)O)ccc(-n2cncn2)c(F)c1 34370,N1(C(C2(CC)CCC2)=O)CC2(CCCC2NC(C2C(C)OC(C)C2C)=O)C1 34371,c1(C(N(CC(CC)NC(=O)CCNS(C)(=O)=O)CC)=O)cc(CO)cc(F)c1 34372,C(=O)(C1CCCn2ccnc21)NC(Cc1cccc(OC)c1)(C)C 34373,c1(CC(=O)NCC(CC)NC(=O)COc2ccsn2)csc(C(C)(C)C)n1 34374,CCCCC(CC)(c1nnnn1CCCSC)NCC1CCCC(CO)C1 34375,c1(NC2(CNC(=O)CC3(C(F)(F)F)CCC3)CCOC2)ccn2ccnc2n1 34376,c1(C(=O)NC2(COC)CCN(C(c3cnn(C)c3N)=O)C2)cc(C)cnc1C 34377,c1(C(N2C(CC)C(NC(c3cnn(CC)c3C)=O)CC2)=O)ccc(=N)[nH]c1Cl 34378,N1(C(c2ccccc2)=O)CCN(C(c2cnc(-c3ccccn3)nc2)=O)C2CC12 34379,C1(CNC(CC2CC(SC)C2)=O)CCCCC1NC(c1nnccc1C)=O 34380,N1(C(C2(CC=C)CCCCC2)=O)CC2CC(CNC(C3C=CCCC3)=O)C2C1 34381,c1(C(=O)NCCC(=C)CNC(c2ncccc2C)=O)nn(C)nc1Br 34382,C1(CNC(c2n(CC)nc(C)c2)=O)CCCCN(C(C23CC(C)(C2)C3)=O)C1 34383,c1(CC(=O)NCC2C(NC(C(c3ccccc3)OC)=O)COC2)ccncc1C 34384,C1(CS(=O)(=O)NCCc2nnc(CC3CCC(C#C)C3)n2N)CCCCN1N=O 34385,CC(C)CCCCCCC(=O)N1CCC2C(NC(=O)C(O)CN(C)C)C2C1 34386,c1(N2CC(C(=O)NC)OCC2)ccc(S(=O)(=O)NCc2csc(Br)n2)c(Cl)c1 34387,C=CC(F)(F)C(=O)N1CC(OC2CCN(C(=O)C=C(C)Cl)CC2)C1 34388,Cc1cc(Cl)cc(C)c1OCC(=O)NC(C)CCCNC(=O)CSc1cccs1 34389,CCC(C)CCC(=O)NCC(C)(CO)NC(C12CC(C)(C1)OC2C)=O 34390,C(=O)(NNC(=O)C(O)c1ccccc1OC(F)(F)F)c1c(C)cccc1Cl 34391,C(=O)(C(CCNC(C1CC1CCOC)=O)OC)N1CC(=CCCC)C1 34392,C(=O)(CCCCC(=O)NCC1(C)CCN(C(c2cnccn2)=O)C1)OC 34393,c1(C(N(C2CCCC2)CCNC(CC#N)=O)=O)ccncc1C(F)F 34394,N1(C(CSC)=O)CCN(CC2CCCN(C(=O)C(C)CF)C2)CC1 34395,CCC(CNC(=O)C(=O)Nc1cc(Cl)ccc1C(F)(F)F)CC(F)F 34396,C1(C(=O)NCC(C=C)(C)C)CN(C(=O)CCc2ccnn2C)CC1F 34397,N1(C(CC=C)=O)CC(C)(C)CCC1CNC(c1cccc(OCCOC)c1)=O 34398,c1(CN(C)CCN(C)C(c2cc(-c3ccccc3)[nH]n2)=O)noc(C2CCC2)n1 34399,CN1CCOCC(NC(=O)CCOCCNC(=O)CC2CCCN(C)C2)C1 34400,c1(C(N2CC(NC(COCCCCC)=O)C(OC)C2)=O)cncc2n[nH]cc12 34401,C1(C(=O)NCC2N(C)CCN(C(C(C)S(N)(=O)=O)=O)C2)CCc2nncn2C1 34402,C1(C)(NC(C=CCOCCOC)=O)CCN(C(=O)CCc2cc(Cl)no2)C1 34403,C1(OC)C2CCN(C(c3cncc(C)c3)=O)C2C1(C)C 34404,C1(OC(C)=O)CCN(C(C2CC(NC(c3ccns3)=O)C2)=O)C1 34405,C1(NC(c2cc(C)c(Br)o2)=O)(CO)CCCN(C(c2nonc2N)=O)C1 34406,c1(CNC(C(n2cc(CCOC)nn2)C)=O)cccc(C#N)c1 34407,C12(C(=O)NC(C)C)CCN(C1)S(=O)(=O)C2 34408,c1(OC)cc(C)c(C(N2CCC(C)(CCNC(C3CCC(=O)N3)=O)C2)=O)c(C)c1 34409,C1(F)(C(N(CCCNC(C2(OC)CCC(C)C2)=O)C2CC2)=O)CC2(CCC2)C1 34410,Cc1ccc(NC(c2cc(C(=O)O)c(C)[nH]2)=O)c(N(C)C)c1 34411,N1(C(C2C(CCOC)C2)=O)CCC(C)(C)C1CC(N1CC(S(C)=O)C1)=O 34412,c1(C(=O)NC(C(C)NC(C=C(COC)C)=O)(C)C)cc(F)c(F)c(O)c1F 34413,c1(C(=O)NC(C(=O)N(CC#C)CC)C2CCCO2)c[nH]c(=NC)s1 34414,c1(C(=O)NC2(CC(=O)N(CC(CCC)O)C)CC2)c(C)n[nH]c1C 34415,Cc1c(Cl)ccc(C(C)(C)C(=O)NCC2CC(NC(C3(C#N)CC3C)=O)C2)c1F 34416,S(=O)(=O)(CC(=O)N1CC(C(C)NC(=O)C(C)N2CCC2)C1)NCC 34417,N1(C(C(C(C)C)C)=O)CCC(CNC(c2ccccc2CO)=O)C(C)C1 34418,c1(CCC)c(C(=O)N(CCCOCCNC(=O)C=C2CCC2)C)cnn1C 34419,C(=O)(C(C)(CC)NC(C)CCC1C(c2ccccc2)CC1O)NCCC#CCC 34420,C(=O)(C(O)CN(C)C)NCCN(C(C)C)C(c1csc(-c2ccccc2)n1)=O 34421,c1(CCC)cc(C(=O)NC(C)CC(C)NC(c2cccnc2F)=O)nn1C 34422,N1(C(c2scc(C(C)=O)c2)=O)CCC(C2CN(C(=O)CC3CCCCO3)C2)C1 34423,c1(C(N(C)CC2CCN(C(CNS(NC)(=O)=O)=O)C2)=O)cnc(O)c(C)c1 34424,N12CCCN(CC1)C1CCN(C1)C(=O)C2.Cc1ccccc1NC(=O)C(C)(C)Br 34425,N1(C(c2cc(OC)n(C)n2)=O)CCN(C(C2CCNC2=O)=O)C(C2CCCC2)C1 34426,Cc1ccc(N2CCCC3(CC(NC(=O)Cn4ccnn4)C3)C2)c([N+](=O)[O-])c1 34427,c1(C(=O)NCC(CO)NC(c2n(CC)ncc2)=O)c(F)cc(C)cc1F 34428,CC(C)CC(F)(F)C(=O)N1CCC(C2CCCCN2C(c2c[nH]nc2[N+](=O)[O-])=O)C1 34429,Cc1cnn(C)c1C(=O)N(C)CC1(CNC(C2COCC(C)O2)=O)CC1 34430,c1(C(N(C2CCN(C(c3cc(C)ns3)=O)C2)CCO)=O)nc(=O)n(C)[nH]1 34431,N1(c2nnc(COC)s2)CCC(CNC(=O)C(F)C(F)(F)F)C1(C)C 34432,c1(C(N(CC(=O)NC(C)C(O)C(C)C)CC)=O)ncnc(O)c1F 34433,Cc1ccc(O)c(C(=O)NC(C)(C)CN(C)C(C2CC2(C)C(C)C)=O)n1 34434,C1(NC(C2C(C(=O)OC)C2)=O)CN(C(c2ccnc(Cl)c2O)=O)CCC1C 34435,C1(CNC(=O)COC2CC2)CCC(CNC(c2csc(C(F)(F)F)c2)=O)CC1 34436,CC(C)CCCCCC(=O)NC(C1CCN(C(C2CC(C)N(C)C2)=O)C1)(C)C 34437,c1(C(=O)NCCC(C)N(C(CC2(CC)CCOCC2)=O)C)ccc2cnoc2c1 34438,CC(CN(C)C)CCC(=O)N1CCCC(C(=O)NCC2CC3OC2C2CC32)CC1 34439,C(N=c1nc(C2CCOCC2)[nH]s1)C1CCN(C(C(C(C)C)OC)=O)C1 34440,c1(C(N(CCNC(C(c2cn(C)nc2)O)=O)C2CC2)=O)c(Cl)ccc2c1OCO2 34441,c1(CC)cc(C(=O)N(CC(O)CN(C(=O)C=CC2CC2)C)C)ccc1Br 34442,C1(CC(=O)NCC2COC(=O)C2)COCCN1C(c1ccc(CO)s1)=O 34443,c1(C(=O)NCC2CN(C(c3ccc(C)cn3)=O)CC2C)n[nH]c2ccc(Br)cc12 34444,c1(C(C)NC(=O)NCC(c2ccc(C)cc2)(C)CO)cc(C)cnc1F 34445,C12(C(=O)NCC(CC)NC(C3CCSCC3)=O)CC1COC2(C)C 34446,C12(CNC(c3cc(OC(CC)C)ncc3)=O)CCC1CN(C(=O)C=CSC)C2 34447,c1(C(=O)NCC(CNC(Cc2c(C)nc[nH]2)=O)F)cc([N+](=O)[O-])c[nH]1 34448,CC1(C)CC(C(=O)NC2CCCC(O)C2O)CCN1C(=O)C1=CCSC1 34449,N1(C(COc2ccc(C)cc2)=O)CC2CC(C(=O)N(CCF)C3CC3)(C2)C1 34450,CCC(CC(=O)NC12CC1CN(C(c1cocc1C)=O)C2)c1ccccc1 34451,c1(NC(C)CCNC(C2CCOC3(CCC3)C2)=O)cc(=O)n2ccccc2n1 34452,N1(C(c2c(CC)nccc2)=O)CC(CNC(=O)CNC(=O)CN(C)C)C2(CC2)C1 34453,Cc1cccc2nc(C(=O)NCC3CC3NC(=O)C=Cc3nccs3)cn12 34454,N1(C(c2cnc(C(C)OC)s2)=O)CCCC(CCNC(=O)COCCO)CC1 34455,C1(C2=CCCCCC2)(C(=O)NC(CNC(C=Cc2cccc(C)c2)=O)CO)CC1 34456,Cc1cc(CNC(C(N2CC(C(F)(F)F)C(C)C2)=O)=O)ccc1F 34457,c1(OCCCNC(C(=O)NC(c2cccc(C)c2)CO)=O)cc(C)ccc1CO 34458,Cc1oc(C(F)(F)F)nc1C(=O)NCC(c1ccc(F)cc1)N 34459,C1(C(=O)NC2CC(OCC(=O)NC(c3ncc(C)[nH]3)C)C2)CCC2(CC2)C1 34460,N1(C(CCC#C)=O)CC(C(=O)NC(CO)C2(O)CC2)CCC1C 34461,C(=O)(CS(=O)(=O)CCO)NC1C2CCN(C(CC3CCC(C)(C)CO3)=O)CC21 34462,c1(CNCc2nnc(N(C)C)o2)c(Br)ccc(Br)c1N 34463,C(C(C)(C(C)C)NC(c1ccc(CC)nc1)=O)NC(CC1(CC=C)CCCC1)=O 34464,CC1CC(C)(C)CCC1NCCC(C)(c1nnnn1C1CCC(F)(F)CC1)SC 34465,O=Cc1cc(F)c(F)cc1NCC(=O)N(CCOc1cccc(F)c1)C1CC1 34466,c1(OC)cc([N+](=O)[O-])ccc1CCN=C(NCC1CC1C)NCC(C)OC 34467,c1(C(N(CC(CNC(COC)=O)O)C)=O)ccc(Oc2ccc(SC)cc2)cc1 34468,C12(C(=O)NCc3cn(C4CN(C(CSCC=C)=O)C4)nn3)CCCCC1C2 34469,c1(C(N2CC(C)C(NC(=O)CCC3CC3(Cl)Cl)C2)=O)csc2c(O)ccnc12 34470,N1(C(C(CC)(F)F)=O)CC2CC(O)C1C2NC(c1cc(C(F)F)ncn1)=O 34471,c1(C(CNC(C2(C(C)C)CC2)=O)NC(C2CC(C)(C)CO2)=O)ccc(F)cc1F 34472,N1(C(C2CC2C2CCCCC2)=O)CCC(C#C)(C2CC2)CC1.C12(OCCO1)CN2 34473,C1(C(=O)NCCC2CCCCC2)COCCN(CC2CCC(F)(F)C2)C1 34474,N1(C(CC(C)O)=O)CC2CCN(C(=O)C=CC3CCOCC3)CC12 34475,N1(C(C2(C)N(C(CN(C(=O)OC)C)=O)CC=C2)=O)CCC2(CC1)CC2 34476,C1(F)(CNC(CC2CC(C)C2)=O)CC(NC(=O)CNC=O)C1 34477,Cn1nc(C(F)F)c(CN2CCC(O)CC2C(=O)Nc2cncc(F)c2)c1Cl 34478,CC(COc1ccccc1)C(=O)N(C)CCN(C(=O)C(C)(C)c1cscn1)C 34479,C#CCC(C)(C)C(=O)N1CCN(C)C(C(=O)N(C)CCC2CCOCC2)C1 34480,c1(OCC(=O)NCCN(C(=O)CC2CCC(=O)O2)C2CC2)ccc(Br)cn1 34481,c1(N2CCCC(C(C)NC(=O)C=CBr)C2)cc(Cl)nc(-c2ccccn2)n1 34482,N1(C(CC(CC)(C)C)=O)CCCN(C(c2cnccn2)=O)CC1C(C)C 34483,c1(C(=O)NCC2CN(C(=O)Cc3ccoc3)CCO2)cc(Cl)cc(Br)c1 34484,c1(N(c2nnc(C(=O)OCC)s2)C)ncnc2c(C)csc12 34485,Cn1cc(C(=O)NCC(C)(C)CC2CN(C(c3n[nH]cc3C3CCC3)=O)C2)nn1 34486,c1(N2CCN(C(=O)NC(C3CCOC3)C#C)C2)ccc(F)cc1OC 34487,C1(CC(=O)NC2CN(C(c3c(C)cc[nH]3)=O)C(C)C2)CC2(CCCC2)CO1 34488,C1(F)(CNC(c2ccn(C3CCCCC3)n2)=O)CN(C(C2CC2(F)Cl)=O)C1 34489,N1(C(CN(C(C(C)C2(O)CCC2)=O)C)=O)CCN(C(C2COCC2(C)C)=O)CC1 34490,c1(CNC(C2(OC)CNC2)C)ncc(C(C)(C)C)[nH]1 34491,c1(CC(=O)NCC(CCOC)NC(CC2CC(OCC)C2)=O)ncccc1C 34492,c1(C(=O)NC(CNC(CC(CC)SC)=O)C)ccc2c(c1)CCN2C(C)=O 34493,N1(C(CCOCC#C)=O)CCC(CNC(=O)CN(C)C2CC2)C12CC2 34494,C1(N(C)Cc2ccccn2)CC2CC1CN2C(c1ccc(Br)cc1)=O 34495,CCCC(C(=O)N1CCC(NC(=O)CNC(=O)C(C)(C)C)C12CCC2)C(C)C 34496,C1(CCNC(C(C)Oc2ccc(Cl)cn2)=O)CC(F)(F)CN1C(c1ccns1)=O 34497,C(=O)(C1=CCC(NC(=O)Cc2ccns2)C1)NC(C)CC(F)(F)F 34498,CC1CN(C(=O)CC=CC(C)(C)C)CC1CCNC(c1nc(Cl)cs1)=O 34499,N1(C(CC(C)(F)F)=O)CCC2(CCC(CNC(=O)C=Cc3cscn3)O2)CC1 34500,C1(NC(c2cc(C)c(F)nc2)=O)CCC(F)(F)C(C)(C)C1 34501,CC1C(NC(=O)C=CC2CCOCC2)CCCN1C(C1CC2(CCC2O)C1)=O 34502,C(=O)(C(C(=O)N1CCC(CN(C(=O)C(C)=C2CCC2)CC)CC1)OC)OCC 34503,C(=O)(CCCCC(C)C)N1CC2C(S)C2C1.Cc1ccc(C2CNCCO2)cn1 34504,c1(C(N2CC3C(NC(=O)CC(C4CC4)C4CC4)(CC3)C2)=O)cn2c(n1)CCCC2 34505,C1(NC(CCC=C=C)=O)CCC2CCN(C(c3ccc(F)c(C)c3Cl)=O)C1C2 34506,c1(CNC(=O)NC(c2ccc(C#N)s2)C(F)(F)F)cc(Br)ccc1F 34507,c1(NC(c2cc(-c3cccc(C(C)=O)c3)[nH]n2)=O)ccc(Cl)c(CO)n1 34508,C(CNC(=O)CC1CCCC1C)(CCNC(C1(C(C)C)CCC1)=O)OC 34509,CC(O)C(F)(F)C(=O)NC1COCC1NC(c1cc([N+](=O)[O-])n[nH]1)=O 34510,N(C(=NCC1=CCCC1)NCC1(C#N)CCC1)CC1N(CC)CCC1 34511,C(=O)(C(C)(C)C(C)O)NCC(C)NC(COCc1c(C)ncs1)=O 34512,N1(C(C(C)SCC)=O)CC(NC(c2nocc2C(C)(C)C)=O)CC1(C)C 34513,N1(C(C2CCC(C)O2)=O)CCN(C(=O)C=CC=C(Cl)Cl)CC1c1cccnc1 34514,N1(C(CN(C(c2c(CCC)n[nH]c2)=O)C)=O)CC(N(C)C)C(C)C1 34515,Cc1ncc(C(=O)NC(C)(C)C(=O)NCCC2CCCCO2)cc1C#N 34516,N1(C(c2cc(C)c(F)cn2)=O)CCC2OCCN(C(=O)CC3CCCOC3)C2C1 34517,c1(CNC(=O)Nc2c(Cl)ccc(C(=O)NC)c2)nn(C)cc1[N+](=O)[O-] 34518,C1(CN(C)C(C2CC(C#N)C2)=O)CCCN(C(=O)C(O)CF)C1 34519,N1(C(CC2CC(C)(C)C(=O)N2)=O)CCC(S(=O)(=O)C(F)F)C1 34520,C(=O)(CCC(C)NC(c1c(Br)noc1C)=O)OCC 34521,c1(NC(C2C(O)CCN(CC#CC)C2)=O)ccc(N=Nc2ccccc2)cc1 34522,C1(C(=O)Nc2ccn3cncc3c2)CN2CC3CC2(CO1)C3 34523,n1(C(C)C)cncc1C(=O)N(CCCNC(=O)CC1CCCO1)C 34524,N1(C(c2cc(OC)cc(C)c2)C(=O)NC(CC)C)CC(C)c2ccccc21 34525,c1(CNC2CC(OC)C(CO)C2)cnc2ncccn12 34526,N1(C(C2CCN(CC)C2)=O)CCCC(NC(=O)CSc2cc(F)ccc2F)C1C 34527,[N-]=[N+]=NC1CCC2(C(=O)NC(CNC(=O)Cn3cnnn3)CO)CC12 34528,N1(C(c2cc(C(C)C)n(C)n2)=O)CCCC(C2CC2NC(C2CC=CCO2)=O)C1 34529,C1(CNC(c2oc(CC)c(C)c2)=O)CN(C(=O)C(CC(C)C)N(C)C)CCCO1 34530,c1(C(=O)NCC2CC(OC)CN2C(c2csc(C(F)F)c2)=O)nnc(O)cc1O 34531,O=S(=O)(c1ccc(F)s1)Nc1ccc(OCC(F)F)nc1 34532,c1(OCC(=O)NCCC2CCC(NC(=O)C3=CCC3)C2)cccnc1 34533,C=CC(C)(CCOC)C(=O)NCCN(C(=O)C1=COCCO1)C 34534,c1(C(=O)NCCCC(C)NC(C2CC3CCC(C2)O3)=O)cccc2c1ncn2C 34535,C(C(O)CC(=O)NCC1CC12CC2)NC(=O)CCc1ncccn1 34536,C1(N(C(CC(C)CF)=O)C)CCC2(CC1)CCN(C(c1ccc(F)cc1O)=O)C2 34537,c1(C(N2C(CNC(Cn3c(C)nnn3)=O)CC2)=O)ccccc1-c1ccccc1 34538,C1(NC(CC(c2ccc(C)cc2)C)=O)CCN(C(C2(C)CCC2)=O)C12CCCC2 34539,CC1(C)NC(=O)CC1C(N1CCCC(C(=O)NC2CC(C)C2)CC1)=O 34540,CC(C)CC(CNC(=O)CCCC#N)C(=O)NCCCC1CC1C 34541,CC(C)CC(C)CC(C)C(=O)NC1(CN(C(=O)CCc2cncnc2)C)CC1 34542,C1(N(C(COCC=C)=O)C)CC2CCC(C1)N2C(C1(C(F)F)CCOCC1)=O 34543,C(=O)(CC(C)(C)C(F)(F)F)NCCOC1CN(C(C(CC)(O)c2ccccc2)=O)C1 34544,c1(CC)ccc(C(N2CCC(C)(CNC(=O)C(O)C(C)C)C2)=O)c(C)n1 34545,C1(CNC(C(C(C)C)OC)=O)CN(C(c2c(C)cc(O)cc2C)=O)CC(C)(C)O1 34546,c1(C(=O)NCC2C(C)CN(C(C3CCCCO3)=O)C2)cc(Br)c(F)cc1N 34547,CCCN(NC(=O)c1ccc(I)cc1OC)C(=O)C1CNC1 34548,C1(CCC#C)CCCN1C(=O)C(C1CCN(C(C2CC(=O)C2)=O)C1)C 34549,N1(C(c2ccc(COC)s2)=O)CCCCCC1CNC(=O)C(C)C(C)C 34550,c1(CN(C(C2CCC2NC(=O)CC2CCCSC2)=O)CC)ccccn1 34551,CC1(CCO)CCN1C(=O)C(c1ccco1)NC(C1CC(CF)C1)=O 34552,Cn1ncc2ccc(CN3CCC(O)(C(=O)Nc4cc(C#N)ccc4Br)C3)cc12 34553,c1(C(=O)NCC2CCC(CNC(C3(C)CC(=C)C3)=O)CC2)cc(N)cnc1C 34554,C1(NC(c2coc(C3CCC3)n2)=O)COC2(C1)CN(C(c1cc[nH]n1)=O)C2 34555,C1(NC(CC(COC)C)=O)CC1C1CCCN(C(c2cnn[nH]2)=O)C1 34556,N1(C(c2ccsn2)=O)CCCC(C2CCN(C(c3conc3C3CC3)=O)CC2)C1 34557,C(=O)(C(CC1CCCC1)C(C)C)NC1CC(NC(c2c(CC)n(C)cc2)=O)CC1O 34558,N1(C(C2C(OCC)C2)=O)CCC(NC(=O)CCn2cccnc2=O)C(CO)CC1 34559,C1(NC(C2C(CNC(c3cccc(=O)o3)=O)C2)=O)C(O)C2CCOC12 34560,c1(OC)cc(OC)cc(CNC(C2CC3CCC2CC3)=O)c1 34561,C12(CNC(c3cc(CC)n(C)n3)=O)CC(CO1)N(C(=O)C(C)CO)C2 34562,C(=O)(CCCC(C)CC)NC1(C(N2CCCCC(CCC)C2)=O)CCOCC1 34563,c1(C(N2CCC(O)(C(C)NC(=O)CC3CC(F)C3)C2)=O)n[nH]c2c1CCC2 34564,c1(C(N(C)CCN(C)C(C2CCCS(=O)(=O)C2)=O)=O)cncc2n[nH]cc12 34565,C=Cn1ncc(C(=O)NC2CC(C(=O)Nc3ccc(O)c(OC)c3)C2(C)C)c1N 34566,C1(C#CC(=O)N2CC(NC(C3(C(C)(C)C)CCCCC3)=O)CC2C)(CC)COC1 34567,C1(C2CC2)(NC(CCNC(c2nn(C)c(O)c2)=O)=O)CCOC1 34568,c1(OC)cc(NCC(C2CC2)N(C(=O)C(C)CC(F)F)C)ccc1[N+](=O)[O-] 34569,CCC(CC(=O)NC1(CCC(=O)NCc2cn(C)cn2)CCCC1)C(C)C 34570,N1(C(C(C)O)=O)CCC(n2cc(CN(CCC(F)(F)F)CC(F)(F)F)nn2)CC1 34571,C1(OCc2cn(CCCCC)nn2)CCCN(C(=O)CC2CCCC(O)C2)C1 34572,C=CC1CN(C(c2ncsc2C)=O)CC1NC(=O)C(C)C1CC1 34573,C1(NC(c2c(C)ccn2C)=O)CC2(C1)CC(C(=O)NCC(c1ccnn1C)O)C2 34574,CC1(C2CC2C(N2CCCC2C(C)(C)C(N2CC3CCC2CC3)=O)=O)COC1 34575,n1(CC(=O)OC(C)(C)C)cc(C2CC(F)(F)C2)nn1.CN1CC1 34576,C(=O)(CC(CC)CCCC)NC(CC#C)CC(=O)NCC1(C)CC(C)C1 34577,CCC(CC(=O)NCC1(C(=O)NCc2ccco2)CCCO1)C1CC1 34578,Cc1nn2cc(C(N3CCC(N(C(=O)C(c4ccccc4F)C)C)C3)=O)nc2s1 34579,N1(CC(N2CCC(NC(=O)CC3CCSCC3)C2)=O)C(=O)CNC1=O 34580,N1(C(c2c(SC)nccn2)=O)CCC2(CCC(NC(c3nccn3C)=O)CC2)C1 34581,CC1C(NC(=O)C(CCN(C)C)NC(c2nc[nH]n2)=O)CCCN1C 34582,n1(CCC)cc(CN2CCC(C(=O)OC)C2)cn1.N12CCC1(C)C2=O 34583,C1(CC)CCC(C(N2CCC2CC(=O)NCC(C)O)=O)CC1 34584,C(=O)(C1=Cc2ccccc2C1C)NC(C)CCCNC(=O)C1=C(Cl)CC1 34585,Cc1ccc(C(N2CC=CC(NC(=O)C(c3ccccc3)O)C2)=O)cc1F 34586,Cc1cc(C(N2CCOC(C(=O)NCCCCC3CCCC3)C2)=O)c(C)s1 34587,N1(C(c2cc(C)ncn2)=O)CCC(CO)C(NC(c2csc(C(F)(F)F)c2)=O)C1 34588,C(=O)(C1=CS(=O)(=O)CCC1)N1CCC(N(C(=O)C(C)CF)CC)CC1 34589,c12cc(Cl)c(c(Cl)c1)[nH]c2=O.c1(-c2c(O)nccc2)c(F)cc(F)cc1F.CO 34590,c1(CC(N2CCCC(CNC(CCc3ncc(C)[nH]3)=O)C2)=O)ccc(F)cc1F 34591,N1(C(C2CCCCC2)C(=O)NC(CC)(C)C)CCSC(Cn2cccn2)C1 34592,C1(C(N(C(C)C(N2CCC2(C)CCO)=O)CC)=O)CCC(F)C1 34593,N1(C(C)C(=O)N2CC(CCNC(=O)CCc3nncs3)C2)CCN(C)CC1 34594,c1(NC(N2CCC(C)(c3cn(CC4CC4)nn3)C2)=O)cnc2ccccc2c1 34595,C1(n2cc(C(C)O)nn2)CCCN(N2CC(CCOc3ccccc3)C2)C1 34596,N1(C(=O)Cc2c(C)cnn2C)CCCC(C)C1CCNC(c1c(OC)scc1)=O 34597,c1(C(=O)NC2(CNC(=O)CCF)CCC2)cc(Cl)c2c(c1)OCCCO2 34598,N#Cc1ccnc(N(Cc2cnn(-c3ccccc3F)c2)CC2CCNC2)n1 34599,c1(C2C(NC(N3C(C=C)CC3)=O)C2)cccc2cnccc12 34600,C=CCC(CNC(C1C2CCCC12)=O)C(=O)N1C2CCC1CC2 34601,c1(CC(N2CC(NC(C=CS(C)=O)=O)CC2(C)C)=O)ccc(Br)cc1C#N 34602,CCCCC(C(=O)NCCCCCNC(c1ccnc2ccsc12)=O)C(C)C 34603,NS(=O)(=O)CC(=O)N1CCCCC1c1n[nH]cc1C(=O)NCC1CCC(O)C1 34604,C12(CNC(C3C(CCC)C3)=O)CC1CN(C(=O)Cc1cncc(Br)c1)C2 34605,C1(C(N2CC(COC(C)=O)C2)=O)C=CC(NC(=O)C(CO)Nc2c[nH]nc2C)C1 34606,Cc1cc2cccnc2nc1C(=O)NC1CN(C(c2cnc(S)[nH]2)=O)C1 34607,C1(NC(Cc2c(C)ccs2)=O)CCCN(C(c2ccccc2C(F)(F)F)=O)C1C 34608,C1(NC(C2N(CC)CC2)=O)CCSC12CN(C(C1CCN(CC3CC3)CC1)=O)C2 34609,c1(SCC(N2CC(NC(c3ccnn(C)c3=O)=O)C2)=O)ccc([N+](=O)[O-])cc1 34610,N1(C(c2cccc(OC)c2C)=O)CCC2C(C1)CN2C(=O)C(C)n1cccn1 34611,Cc1cc(NC(C2CN(C(=O)C(c3cncnc3)C)CC2C)=O)c(C)cc1O 34612,C1(NC(C=CC(=O)OCCCC)=O)CC2(C1)CN(C(C1(C)CCC1)=O)C2 34613,N1(C(CC(C(C)C)C(C)C)=O)CCc2c(c(CNC(C3CC3F)=O)nn2C)C1 34614,c1(C(=O)NCCCC(C)NC(C2CN3CCC2CC3)=O)nn(C)c2c1CCCC2 34615,c1(CC(N2C(C)CC(Nc3nccc(CO)n3)C2)=O)cn2ccccc2n1 34616,C(=O)(CC(F)(F)CC)NC(C(C)NC(C(CCC)NC(=O)OC(C)(C)C)=O)CO 34617,Cc1cnc(N)c(C(=O)NC2CC(CNC(c3cccc(Cl)c3F)=O)C2)c1 34618,Cc1nn2cc(C(=O)NCC(CC(C)C)NC(C3COC(=O)N3C)=O)nc2s1 34619,C#Cc1cccc(C(N2CCN(C(c3cc(C)nnc3O)=O)C(CCO)C2)=O)c1 34620,N1(C(=O)CCC2CCCCN2C(c2cncc(O)c2)=O)CC2CCCC(O)C2C1 34621,CC1CCN(C(c2cn(CC3(C)COC3)nn2)=O)CC1NC(c1cnn(C)c1)=O 34622,N1(C(C(CC)N(C)C)=O)CC2CCC1CN2C(=O)CC1CCOC1 34623,c1(C(N(CCNC(c2nc(C(C)(C)C)sc2)=O)CC2CC2)=O)cc(C2CC2)ncn1 34624,c1(OC)ccccc1C(=O)NCC(C(C)C)NC(c1cnn(C(F)(F)F)c1)=O 34625,N1(C(=O)OC(C)(C)C)CC2CCCN(Cc3cccc(F)c3Cl)C2C1 34626,c1(C(CC(=O)N(C2CCN(C(=O)COCC3CC3)CC2)CC)C)ccc(F)cc1 34627,C(=O)(C(C)(C)CCC(=O)NCC(C)CNC(C1CC2C=CC1C2)=O)OC 34628,CCC(O)C(C)C(=O)NC1(CO)CN(C(=O)C=CC(C)C)C1 34629,Cc1ocnc1CC(=O)N(CCCCCNC(=O)CC(C)n1cccc1)C 34630,C(CCCC(C)NC(=O)CCCc1ccsc1)NC(C1C(C(C)=O)COC1)=O 34631,C(C(=O)N(CC(C)CNC(c1ncoc1Br)=O)C)(C(C)C)SCC 34632,c1(C(C)N(C(c2ccc(O)cn2)=O)C2CC2)cccc(S(N)(=O)=O)c1 34633,C1(NC(C)=O)CCCCC12CCN(C(c1cc3c(Cl)cc(F)cc3[nH]1)=O)C2 34634,c1(NC(=O)OCC)ccc(C(=O)NCC2CCC(NC(=O)C(C)O)C2)cc1 34635,c1(C(N(CCNC(=O)C(C2CCCO2)OC)CC)=O)cc(C)ccc1OC 34636,n1(CC(=O)OC)cnc(C)c1C(=O)N(CCCNC(=O)C(C)Cn1ccnc1)C 34637,N1(C(c2ncn(CC)n2)=O)CCC2CC12C(=O)NCCCc1c[nH]nc1C 34638,C1(C(=O)NCCOC2CN(C(CC3(C=C)CC3)=O)C2)CCS(=O)(=O)C(C)C1 34639,N1(C(C23CC(OC)C2C3)=O)CC(NC(c2cc(C(C)C)on2)=O)C(O)C1 34640,CC(=O)CCN=C(NCCCCCF)N1CCC(C2CC2)C1 34641,N1(Cc2c(OC)cccn2)C2CCCC1CC(NC(C1(C)CCCC1)=O)C2 34642,c1(OC)cc(C)c(C)cc1C(N1CCC1(C)C(=O)Nc1sccc1C(N)=O)=O 34643,CC(C)(CCNC(C1CCC1C(C)(C)C)=O)NC(=O)OC(C)(C)C 34644,Cc1cc(CCN2CCC(C)C2c2cccc(C(F)(F)F)c2)ccc1OC(F)F 34645,C(C(C)(C)CCNC(CC(C)C1CCCO1)=O)NC(C1(CO)CCOCC1)=O 34646,C1(CCOCCC(=O)NCC(C)N(C)C)CCCNC1 34647,N1(C(CCOCCOCC)=O)CC(O)CC1C(=O)N(C1CCC(OC)CC1)C 34648,c1(C(N2C(C)CC2C(=O)NC2CCCCC2)=O)ccn2cncc2c1 34649,c1(CC(=O)NC2CCN(C(C(CC)F)=O)C2(C)C)ccc2nc(O)[nH]c2c1 34650,N1(C(c2cc(COC)on2)C(=O)NCCCC)CCOC(c2n[nH]c(C)n2)C1 34651,C1(CC(=O)NCC2C(NC(C3CN(S(CC)(=O)=O)C3)=O)C2)CCC(F)(F)CC1 34652,CC(C)CC(F)C(=O)NC1CCCC1NC(c1nn(C)cc1Br)=O 34653,Cn1cnc(C(N2CCCCC2CNC(C2CCCC2(C)C)=O)=O)cc1=O 34654,C12(NC(c3ccc(O)nc3)=O)CCCC1N(C(c1ccc3nccn3c1)=O)CC2 34655,N1(C(c2c(C)nc[nH]2)=O)CCOC(C(C)NC(=O)C(F)(F)c2ccsc2Cl)C1 34656,CC1CN(C(C2CCCN2C)=O)CCN1C(c1cc(Cl)ns1)=O 34657,Cc1c(CN(C(N2CCC2C2CCCCC2)=O)CC2CC2)oc2ccccc12 34658,C(=O)(C(CCSC)NC(=O)NC(C)(C)C)NC12CC(OC)C1C2 34659,c1(Cn2cc(CN(C(C(C)OCC=C)=O)C3CC3)nn2)ccc2[nH]ncc2c1 34660,c1(C(=O)NC2CCCN(C(C3C(C(C)C)CCC3)=O)CC2)cnc2c(c1)CCC2 34661,Cn1ncc(=NC(=O)C2CC23CCN(Cc2ccc(C(=O)O)s2)C3)[nH]1 34662,c1(C(=O)NC2CCCC(NC(C3CC(F)C3)=O)C2)c(F)c(F)c(F)c(F)c1F 34663,N1(C(c2cc(CC)n(CCO)n2)=O)CCC2(CCCN2C(=O)C(O)CSC)CC1 34664,Cc1cnc2cc(C(N3CCCC3C(C)NC(=O)CC(F)(F)F)=O)nn2c1 34665,N1(C(C2(COC)CCCC2)=O)CCC(C2CC2)(NC(=O)C(O)C2CCCC2)C1 34666,C1(C2(O)CCOC2)(C(N(C)CC2CCN(C(c3ccc(C4CC4)o3)=O)C2)=O)CC1 34667,C1(NC(C(Cn2cncn2)NC(c2cc(C)n(C)n2)=O)=O)CC(C2CCC2)C1 34668,C1(NC(COCCC)=O)CC2CN(C(C3CC(Cl)(Cl)C3)=O)CC2C1 34669,C1(NC(c2c(C)noc2)=O)CC2CCC1N2C(=O)C=CC1CCOC1 34670,C=CCC(CC(C)C)C(=O)NCc1ccc(C(=O)NC(C)C(C)n2cccn2)o1 34671,N1(C(C(C(C)C)CN(C)C)=O)CCN(C(=O)CCCC(N)=O)C2(CCC2)C1 34672,CC(CC(=O)N1CCC(C(=O)NCC(C)(C)N2CCCC2)O1)N(C)C 34673,C1(NC(C2(CC#C)CCCO2)=O)CCN(C(=O)CN2CC3CC3C2)C1CC1CC1 34674,C1(NC(c2cc(C(C)=O)on2)=O)CCCCC1NC(=O)CCc1cncnc1O 34675,c1(CC)oc2ccccc2c1C(N1CC(CNC(=O)C(C)CSC)C(F)(F)C1)=O 34676,CC(CO)CCCNC(C1COC(CNC(=O)COCCN(C)C)C1)=O 34677,Cc1nc(CC(=O)N(C)CC2(O)CN(C(C3(NC(N)=O)CC3)=O)C2)co1 34678,C(=O)(CCCCBr)NC(CC(=O)Nc1nccs1)c1ccccc1 34679,c1(OC(C)C(=O)NCC2CCN2C(c2nn(C)cc2C(F)F)=O)cccc(F)c1 34680,CCCC(C)CC(=O)NCCC1(O)CCCN(C(c2nc(CC)oc2C)=O)C1 34681,C(=O)(CCCCCCO)NCC1OCCCN(C(C(C)OCC(F)(F)F)=O)C1 34682,c1(C(N(C)CCNC(C2CS(=O)(=O)CC(=O)N2)=O)=O)cccc2cnnc(O)c12 34683,Cc1sc(Cl)nc1C(N1CCCCC1CN(C)C(C1CC1CF)=O)=O 34684,c1(C(N2C(C(=O)OC)CCCC2)=O)cc(=O)n(CC#N)cn1 34685,C1(CC(=O)NCCCN(C(=O)CC=CC=C(C)C)CCC)CCC(C)C1 34686,c1(C(=O)NCCCCCN(C(=O)CC2CC2(C)C)C)cnn2c(Cl)cccc12 34687,Cc1cc(CNC(=O)C(C2CCCO2)NC(c2ccc(C)o2)=O)n(C)n1 34688,CC1CN(C(=O)CSS(C)(=O)=O)CC1NC(=O)CCCc1ccsc1 34689,n1(CC)cc(Cl)c(C(=O)NC2CCC2NC(c2cnc[nH]2)=O)n1 34690,N1(C(c2n[nH]c(C)c2Cl)=O)CCCC(C)(CNC(=O)CC2CC(C)(C)CCO2)C1 34691,N1(C(c2cc(CCC)[nH]n2)=O)CCN(C(C2CCC(=O)N2)=O)CC1C(C)(C)C 34692,S(=O)(=O)(c1c[nH]c2nc(Cl)ccc12)NCC1CCC(CC)C1 34693,C1(CNC(CCNC(=O)OCC)=O)CC2(CCC2)CN1C(C1CC1(Cl)Cl)=O 34694,C1(NC(CCC2N(C)CCC2)=O)CC=C(C(=O)Nc2ccc(C3CC3)nc2)C1 34695,O=S(=O)(c1ccncc1)NC1C2CCC1CC(CO)C2 34696,CC(CS(C)(=O)=O)C(=O)N1CC2CC(NC(c3ccc(N(C)C)nc3)=O)C(C2)C1 34697,C1(NC(=O)C(C2(O)CCCC2)F)CCSC12CN(C(c1ccc(F)cc1Cl)=O)C2 34698,CC(CCC(C)(C)C)N=c1[nH]c(=N)[nH]c(=NCCc2c(N)cccc2F)[nH]1 34699,Cc1cc(C(N2CCC3(C2)CN2CCC(CC2)C(=O)O3)=O)sc1C.C1(CO)CC1 34700,c1(CC(=O)NC(CC)(C)CNC(=O)Cc2cccs2)ccc2scc(C)c2c1 34701,c1(CCC)nnc(S)n1CC(=O)N(C)CC1(NC(c2cc(C#N)cs2)=O)CC1 34702,CCCCC(CCCC)CC(CC)C(=O)N(CC1=CCCOC1)C 34703,C=CCC(C)(C)C(=O)NC1CCN(C(=O)CCCCC2CC2)CC1CO 34704,OC1COC2C(NC3CN(c4nn[nH]n4)C3)COC12 34705,c1(C(CC(=O)NCCOCCN(C(=O)C(=O)C(C)(C)C)C)O)cc(Cl)cc(Cl)c1 34706,CC1CC2(CCO1)CC2C(=O)NCCN1CCN(c2ccncc2[N+](=O)[O-])CC1 34707,N#Cc1ccc(CC(=O)NCC2CCN(C(=O)CCN3CCCC3)C2)cc1 34708,C(c1ccc(F)cc1)=CC(=O)NCC1CC(F)(CNC(C2(F)CC2(Cl)Cl)=O)C1 34709,N(C(=NC1CCCC1)N(C)C1CCSC1)C(c1cccc(F)c1)C#C 34710,c1(CCC(=O)N(CC)Cc2cn(CCN3CCOCC3)nn2)ccc(Br)cc1 34711,N1(CCOCC)CCN(C2CCN(C(=O)CC(N)C3CCOCC3)C2)CC1 34712,C1(CN(C(C(n2ccc(C(F)(F)F)n2)C)=O)C)CC(F)CN1C(c1ccco1)=O 34713,N1(C(=O)NCCCc2cccc(C)c2)CCC(C)(C)C(CO)C1 34714,N1CCC2(CCC(NC)CC2)C1.C(=O)(CCC(=O)C1CC1)Nc1cn(C(C)C)nc1 34715,C1(c2n(C)ccn2)CCCN(C(=O)C(C)(N)C(F)F)CC1 34716,N1(C(c2ccc(OC)c(SC)c2)C(=O)NC2CCCC2)CCOCC12CCC2.C(C)C 34717,C1(C)(C(=O)NC(CC=C)CNC(=O)CN2CC(F)(F)C2)CCCOC1 34718,C(=O)(C1=NNC(=O)CC1)NC1C=CC(CNC(c2c(C(C)(F)F)cccc2)=O)C1 34719,c1(C(=O)NC23C(CN(C(c4ccn(CC#N)n4)=O)C2)C3)cccc2c1CCO2 34720,Cc1c[nH]c(C(=O)NCC(C)(C2CC2)NC(c2cnc(C(N)=O)s2)=O)c1 34721,Clc1ccc(CNc2cnn(C3CCOC3)n2)c(I)c1 34722,N1(C(C2CCC(COC)C2)=O)CCN(C(c2ccc(F)s2)=O)CC(O)C1 34723,C(C(O)CS(=O)(=O)c1cccs1)NC(c1ccc(-n2ncc(C(=O)O)c2)cc1)=O 34724,CC1CCN(C(C2CCC=CO2)=O)CC1NC(=O)CC1CCC(C(C)(C)C)CC1 34725,C12(C(N3C(C)CC(NC(=O)CC4CCC4)CC3)=O)CCCCC1CCCC2 34726,C#CC1CC2CCC1N(C(C1CCN1C(c1conc1CC)=O)=O)C2 34727,c1(C(C(C)(C)C)NC(COCCNC(CC2(OC)CCC2)=O)=O)cccc(C)c1 34728,c1(C(N2CCC(F)(CNC(c3ncn(CC)n3)=O)CC2)=O)cc[nH]c2nccc1-2 34729,c1(C(N2CCC(O)(C(C(=O)NC)(F)F)C2)=O)nc(C(F)(F)F)ccc1Br 34730,n1(CC(=O)NCC2CCCN(C)C2=O)cnc2ccc(F)cc2c1=O 34731,c1(NC(c2nn(C)cc2Br)c2n(CCCSC)nnn2)nnc(C)n1C 34732,C(CCOCCO)(C(=O)N(C(C(N)=O)C1CC1)C)NC(C=CCC)=O 34733,C1(C(N(CC(C)(C)CO)C)=O)(CN(C)C)CCCC1 34734,CCC(CC)(C(=O)NCCCN(c1cc(Cl)ncn1)C(C)C)c1ccccc1 34735,Cn1c(Br)cnc1NC(N1CCN(c2ccc(Cl)nn2)CC1)=O 34736,c1(OC)ccc2c(c1)CCC2(C)CNc1nc(OC)ncc1Cl 34737,C(=O)(C#CC1CCCCC1)N1CC(N(C)C(c2ccc(Cl)c(F)c2)=O)C1 34738,c1(OC)ccccc1C(=O)NC(CNC(=O)C(C1CCCC1)OC)CO 34739,Cn1cc(C(N2CCC(O)(CNC(C3CCC(=O)N3)=O)C2)=O)c2cc(F)ccc12 34740,Cc1cc(C(N2CCC(C)(C(=O)NCC3(C)CC4CCC3C4)CC2)=O)c(C)n1C 34741,C#CC1CCC(NC(c2csc(CNC(c3ccc(CO)cc3)=O)c2)=O)C1 34742,N1(C(C(N2C(CC)CCC2)=O)=O)CCOCC1CN(C(=O)Cc1ccsc1)C 34743,C(=O)(CCC(=O)NN(C)C)NC1C(CO)CCN(C(COCCCC)=O)C1 34744,c1(C(=O)NCC23CC2CN(C(C2CC=CC2)=O)C3)cccc2cccn12 34745,c1(C(=O)NCC(C(C)C)NC(C2CC2C#N)=O)ccc(SC(F)(F)F)nc1 34746,N1(C(C2ON=C(C)C2)=O)CC(NC(=O)C2=CCCSC2)CC12CCCC2 34747,C1(NC(CC(=C)C)=O)C(C)CN(C(=O)CN2CCCCCC2)CC1C 34748,c1(CCCC)ccccc1-n1nnnc1C1(NC2(COC)CC2)CSC1 34749,N1(C(C(C)(C)OC)=O)CCCC2C1CCN2Cc1cc(Br)ncc1Br 34750,c1(CC(=O)NCC2C(NC(C(CC)O)=O)CC2)c(C)nn(CC(C)C)c1C 34751,CC(C)C(CC(=O)NCC1CC1C(C)C)NC(C1CC2CC(=O)C1O2)=O 34752,C(CCC(C)C(=O)NCC1(C(=O)NOCCCO)CCOC1)OC 34753,c1(C(N2C(CNC(C3CC34CCCC4)=O)CC(O)C2)=O)cnn2c1CCC2 34754,CC1(C(=O)NC2(CC(N3CC4(CC4)C3)=O)CC2)CC(F)(F)C1 34755,C1(NC(Cc2nc(C)[nH]n2)=O)CNCCOC1 34756,C1(NC(CC(=C=C)C)=O)CN(C(=O)CC2CCCOC2)C2(CCOCC2)C1 34757,c1(CC)nc(C(=O)N(C2CCCCC2NC(=O)C(CC)n2cccn2)C)c(C)o1 34758,C(C)(C(=O)NC1(C)CCC(C)C1)(C(C)C)NC(C)=O 34759,c1(C(=O)NC2CC(CNC(=O)COC3COC3)C2)cc(Cl)ncc1F 34760,N1(C(CCOCCOC)=O)CCOC(C(C)NC(c2c[nH]nc2C(=O)OC)=O)C1 34761,c1(C(N(C2CCN(C(C3CC34CC4)=O)CC2)CC(C)C)=O)ncncc1Cl 34762,c1(C(=O)NC2(C3CCN(C(=O)C=C4CCC4)C3)CC2)ccc2cnnc(O)c2c1 34763,C(CC(C(=O)NC(c1cncc(F)c1)C)NC(=O)Cc1nc(=N)[nH][nH]1)=CC 34764,c1(C(N2CC(NC(c3n(CC)nnc3)=O)C3C2C3)=O)cnc(N)c(N)c1 34765,Cc1ccc(CNC2CC3(C2)CC(C(=O)NCc2ccc(C#N)cc2)C3)c(O)c1 34766,N1(C(C=C(C)C2CC2)=O)C2COCC1CC(NC(=O)Cc1cnn(C)c1)C2 34767,c1(C2(OC)CC2)nnc(N(C(c2ccc(C(F)(F)F)cc2)C)C2CC2)n1CC(C)C 34768,C1(C(C)C)CN(C(c2cnc(O)o2)=O)CC1C(=O)N(C1CCC(O)CC1)C 34769,c1(OCC(=O)NCC(CC=C)NC(=O)C(C)=CC2CC2)ccc(C(C)(C)C)cc1 34770,C(=O)(C(O)C(C)(C)CC)N1CC(NC(CCC=CCC=C)=O)C2(C1)CC2 34771,C1(C(N(CCN(C)C)CC)=O)(C(=O)NCCc2nonc2N)CCOCC1.C(=O)N 34772,C1(C(C)NC(c2cc(Cl)c[nH]2)=O)CCCCN1C(=O)CCCc1ccccc1 34773,N1(C(C2C(NC(CCOC(C)=O)=O)CC2)=O)CCOC(C#N)C1 34774,c1(C(=O)NC(CNC(c2occ(C(=O)OC)c2)=O)(C)CO)cc(O)nc(C)n1 34775,CN=S(C)(=O)c1cccc(CNC2CCN(C(=O)OC(C)(C)C)CCC2CO)c1 34776,C#Cc1ccc(NC(=O)Nc2ccc(C(=O)OCC)cc2OC)cn1 34777,Cc1ccc2nc(N(CC(O)CNC(=O)C(c3c(C)nn(C)c3C)C)C)sc2n1 34778,CC1(C)OCCOC1CC(=O)NCCOCCCNC(=O)CC1OCCCO1 34779,C12(NC(C(=C)F)=O)CCC(NC(=O)Nc3nnc(-c4ccc(Cl)cc4)s3)(CC1)C2 34780,N1(CC(C)SC)C(=O)CN(CC=CC(F)(F)F)C1=O 34781,C1(CCC(=O)N(C)CCO)CCCN(C(c2cocc2C(N)=O)=O)C1 34782,C1(NC(C2(C)N(C)CCC2)=O)C2CCC(C2)C1C(=O)NC1COCC1O 34783,Cn1cnc(CNc2cccc(OCC3CCCCC3)c2)cc1=O 34784,c1(C(N2CCC(C(N3CCCC(C)C3)=O)CC2)=O)c(Cl)ccc(Br)c1N 34785,c1(C(=O)NCCCCCN(C(=O)CC2CCCC(F)(F)C2)C)cc(=O)n(C)cn1 34786,n1(C(C)C)cncc1C(=O)NCC1CCCC1NC(C1CC(N(C)C)C1)=O 34787,C1(C2CCN(C(C3(C)CC3C)=O)C2)(NC(c2n[nH]c(C)c2C)=O)CC1 34788,c1(C(=O)NCC2(OC)CN(C(C3(CC)CCCCO3)=O)C2)ccc(C)cc1Cl 34789,c1(CN(CCC(=O)OCC)C(=O)NC)ccc(C)cc1OCCCCCC 34790,C(=O)(C(CCC(C)C)NC(c1c(C)n[nH]c1C)=O)N1CC(CC)(CC)C1 34791,N(C(=NCCC(=O)N(C)C)NC1CCOCC1F)Cc1n(CCC)ncn1 34792,C#CCCC(=O)N(CCC(C)(C)NC(C1CC(NC(C)=O)C1)=O)C 34793,c1(OC)ccc(S(=O)(=O)NCC2(F)CCCN(C(=O)CC3CC3)C2)cn1 34794,C(CC(C(=O)N(C)Cc1nc(C)no1)NC(=O)CCCc1ncco1)OC 34795,c1(CC(=O)NCC(C)NC(CC(c2cccc(OC)c2)C)=O)ccc(F)c(C)c1 34796,N1(C2C3CN(C(C(C)(C)CCl)=O)C(C3)C2)CCc2ccncc2C1 34797,C12(NC(N3CCN(C(c4ccc([N+](=O)[O-])cc4)C)CC3)=O)CCOC1CS(=O)(=O)C2 34798,N1(C(C(CC#C)(C)C)=O)CC2CCC1C(CNC(C1(c3ccn(C)n3)CC1)=O)C2 34799,N1(C(c2sccc2Br)=O)CCCC(O)(Cn2cc(C3(F)COC3)nn2)CC1 34800,c1(C(=O)NC(CC(C)NC(c2c(C#C)c[nH]n2)=O)C)noc2c1CCCC2 34801,Cc1nc(O)nc(O)c1CC(N1CCCC(CNC(C2(C(N)=O)CCC2)=O)C1)=O 34802,c1(C(C)=O)ncc(C(N2CC(C(C)(C)O)(CNC(=O)Cc3cnc[nH]3)C2)=O)s1 34803,N(C1CC2(CCC2)Oc2ccc(F)cc21)C(=O)NCCCC(C)CO 34804,C1(C(N2CC(C(C)O)C2)=O)CN(C(=O)CCc2cncs2)CC2(CCC2)C1 34805,c1(C(=O)NCC(C)NC(=O)Cc2ccc(Br)cc2)nccc(C#N)c1F 34806,c1(CCNC(=O)C(=O)NCC2CCCC2O)c[nH]c2cccc(Br)c12 34807,c1(OC)ccccc1NC(C1CCCN(C(C2(C)CC(C)(C)C2)=O)C1)=O 34808,CCCCCCCCC(F)C(=O)OCC.C(=O)C1CCCc2nncn21 34809,c1(C(=O)NCC2CC(NC(CCCCCC#N)=O)C2)ccc2c(O)nncc2c1 34810,C=CC(C)CC(=O)NCCOCCOCCNC(C1CCCCO1)=O 34811,N1(C(CCC(C)OC)=O)CCCC(F)(C(=O)NC2CC(C)C2)C1 34812,C1(CC=C)CCCCN1C(C1CCN1C(=O)CC1CCOC1)=O 34813,N1(C(C(CC)(C)F)=O)CCC2(CC1)CN(C(C1CC(=C3CCC3)C1)=O)C2 34814,O=C(C1=CC(O)CCC1)NCC(C1CCCC1)NC(c1cccc[n+]1[O-])=O 34815,C(c1ccccc1)=C(C(=O)NCC1C(NC(CCC=C)=O)CCC1)CC 34816,n1(CC)cccc1C(c1nnnn1C1CCOC1)NCc1cncs1 34817,c1(C(=O)NC(C(CO)NC(C(C(C)O)N(C)C)=O)C)nnc2n1CCCCC2 34818,Cc1coc(C(C)(C)C)c1C(N1CC(N(C(=O)C(F)C2CCOC2)C)C1)=O 34819,c1(Nc2c(C(=O)NC3(C)CC3)ccc(Cl)n2)cc(Cl)c(F)c(Cl)c1F 34820,N1(C(C2(C)N(C(c3c(CC)noc3)=O)CCC2)=O)CCc2ncncc2C1 34821,C1(C(=O)NC(C)CNC(=O)CC2(C)CC(F)(F)C2)CC2(C1)C(F)(F)C21CC1 34822,C(CO)(CC(F)(F)F)NC(C(c1n(C)ncc1)NC(C1OCCC1(C)C)=O)=O 34823,C(=O)(CC1=CCN(C(C23CCC(OC)C2C3)=O)CC1)N(CCC=C)CC 34824,C1(CCNC(c2coc(Cl)c2)=O)CCCN(C(C2CCCCN2CC(F)F)=O)C1 34825,N(C1CCOc2ccc(Cl)cc21)C(=O)NCc1ccc(F)cc1N1CCOCC1 34826,N1(C(c2ccn(C)n2)CC)Cc2cnc(C)nc2C1 34827,C#Cc1ccc(CC(=O)NCC2(NC(c3coc(C(F)(F)F)c3)=O)CC2)cc1 34828,N1(C(c2n(C(CC)C)ncc2)=O)CCN(C(=O)CC(C)(C)C2CC2)CC1C(C)C 34829,CC(C)S(=O)(=O)CCCN(C1CCCN(C(=O)C(=O)Nc2ccccc2)CC1)C 34830,CC(C)(Cc1cnn[nH]1)C(=O)N1CC(NC(C2CCC(O)C2)=O)C(O)C1 34831,c1(CNC(C(C)n2cncn2)=O)cc(C(=O)NCC(C)(C)C2CCCO2)on1 34832,c1(C(CNC(=O)NCC(COCCC#C)(C)C)N(C)CC)ccc(Cl)cc1 34833,S(=O)(=O)(c1ccncc1)NCC1CCN(C(=O)Nc2ccc(F)cc2)CC1F 34834,CC1c2c[nH]nc2CCC1C(N1CCC(CNC(=O)CC2=CCCC2)C1(C)C)=O 34835,N1(C(C(CCC)NC(C)=O)=O)CCN(Cc2cnc(OC)c(C)c2)CC1C#N 34836,c1(C(=O)NC(C)C(=O)NC(c2nc[nH]n2)CO)cc[nH]c2nccc1-2 34837,c1(N2CC3C(CNC(CSCC#C)=O)C3C2)ccc([N+](=O)[O-])c(C)n1 34838,C1(C(N2CCN(C(CSCC#C)=O)C(CO)C2)=O)OCC2COCCC12 34839,c1(C(=O)NCC(CC)NC(c2snnc2C)=O)cccc2cnsc12 34840,C1(NC(c2nc(C(=O)NCC3CC(O)(CNC(C)=O)C3)sc2)=O)CC2(CCC2)CO1 34841,Cc1ccc(NC(=O)CN(C2CCN(C(c3ccc(CON(C)C)o3)=O)C2)C)cc1 34842,c1(C(=O)NC2C(SC)CN(C(=O)CN3CCSCC3)C2)nccn2cc(C)nc12 34843,N1(C(=O)CCN2CCCC2)CCC(C(N2CCCC(CN(Cl)Cl)C2)=O)CC1 34844,C1(C(N2CCN(CCN(C(=O)Cn3ccnn3)C)CC2)=O)CCCC12OCCO2 34845,C1(CC(C)NC(C(=O)N(CCC(=O)NCC2CC2)CC)=O)CCCCC1 34846,N1(C(CNC(CC)=O)=O)CC(NC(=O)Cc2ccccc2C)CCC1C 34847,N1(C(CC2CNC(=O)N2)=O)CCCC2CN(C(c3cnn(CC4CC4)c3)=O)CC12 34848,C1(C(=O)NC(C2CCN(C(=O)CCc3cnc(C4CC4)o3)C2)C)C=CC=CC=C1 34849,C(C(F)(C(=O)N1CC(C)(OC)C1)C(C)C)NC(c1ccc(=NC)[nH]c1)=O 34850,C(=O)(C(CCN(C)C)NC(c1cnnc(O)c1)=O)N1CCC(CC)C1 34851,c1(CC2C(=O)NS(=O)(=O)C3(CC3)c3cn2nn3)ccc(O)cc1.CCF 34852,C1(C(N2CC(C)C(NC(C3(C(C)(F)F)CC3)=O)C2)=O)CC1C1CCOCC1 34853,CCC(CC(=O)NC1CC2(C1)CC2C(=O)N(C)CCn1cnnc1)OC 34854,c1(CCC)nc(C)c(C(=O)N(C2CCCC(NC(c3cn(C)c(O)n3)=O)C2)C)o1 34855,N1(C(NOCC(=O)N(C)Cc2cnn(CC(F)(F)F)c2)=O)CCCCC1=O 34856,C1(CC#C)CCCCN1C(C1CCCN1CCCN(C)C)=O 34857,N1(C(CSC)=O)CCN(C(C2CCCN(C(=O)CC3(C)CC3(Cl)Cl)C2)=O)CC1 34858,Cc1nc(O)c(C(N2CCCC(CNC(=O)CCCCC#N)C2)=O)nc1C 34859,c1(CC)nc(C(C)C)ccc1C(=O)NCCCNC(c1ccn(C2CCC2)n1)=O 34860,c1(C(=O)Nc2ccc(O)cc2Br)ccc2ncc(-c3ccc(F)nc3F)n2c1 34861,c1(C(=O)NCCN(CC(=O)NC(C)COCC)CC=C)ncc[nH]1 34862,N1(C(c2c(OC)nccc2)=O)CCCC(N(c2cnc(C#N)cn2)C)CC1 34863,c1(C(N(C2CCN(C(C3CC3(F)F)=O)C2)CC)=O)c2c(nn1C)CCC2 34864,c1(C(N2C3CN(C(=O)Cc4cn[nH]c4)C(C3)C2)=O)nc2cnccc2s1 34865,C(CC(C)(C)F)NC(C(C1CN(C(=O)CCCNC(C)=O)C1)OC)=O 34866,Cc1cncc(C(=O)NOC2CCN(C(=O)Cc3csnn3)C2)c1 34867,C1(C(N2CCC(NC(CC(C=C)CC)=O)C(C)C2)=O)CCC2(CC1)CNC(=O)C2 34868,CC1(C(=O)NC2CC2NC(=O)C(c2ccc(F)cc2)(F)F)CCC(O)CC1 34869,N1(C(COCC)=O)CCN(C(C2CCCCN2C(=O)CC)=O)CC1CCOC 34870,c1(C(N2CC(C=C)C(NC(=O)COc3cn[nH]c3)C2)=O)csc2ccc(F)cc12 34871,C(CCCCC(=O)NC1CCC(C(N)=O)CC1)N(C(=O)C(=O)C1CCCC1)C 34872,Cn1ccc2sc(C(N3CCCCCC(NC(=O)CN4CSCC4=O)C3)=O)cc12 34873,C1(OC)CC(CC(=O)Nc2ccc(SCCCC(=O)OC(C)(C)C)cn2)C1(C)C 34874,c1(NC(N=c2[nH]n(C(CC)C)c(C)c2)=O)cccc2c1nc(O)n2C 34875,c1(C(N2CC(NC(C3(OC)CCOC3)=O)C(O)C2)=O)c(N)sc(C)c1C 34876,CC1=NNC(=O)C1CCC(=O)NCCCOC1CCN(C(C2CC(O)C2)=O)CC1 34877,c1(CC)c(C(C)NC(c2nn(C)cc2C)=O)oc2ccccc12 34878,C1(NC(c2c(O)ncc(NC(C)=O)c2)=O)CCC2(CCCNC2)C1 34879,c1(C(=O)NC(CC)CNC(C2CN(C(C)C)CCO2)=O)cc(O)ccc1N 34880,CC1CN(C(C2CC2c2ccc(Br)cc2)=O)CCN1S(=O)(=O)c1nccs1 34881,C=CCN=C(NCCC1CC(C(=O)NC)C1(C)C)NCC(C)(C)NC(C)=O 34882,Cc1cccc2nc(C(=O)NC(C)(C)C(C)NC(C3CNC(=O)N3)=O)cn12 34883,c1(C(=O)NCC(CC(C)C)NC(C2(SC)CC2)=O)cnc2ncnn2c1O 34884,c1(C(=O)NCC(C(C)(C)C)NC(c2c(C)cc(CO)o2)=O)cc(C)c(O)c(N)c1 34885,CCC(CC)C(C)C(=O)N1CC2CC2(NC(=O)Cn2nc(C)oc2=O)C1 34886,c1(C(N2CCC(C(C(=O)NC(CCC)C3CCC3)F)C2)=O)cc(OC)n(C)n1 34887,C1(C(N(C(C)CC2CC2)C)=O)C2CC3C(C2NC(=O)C(C)C(F)F)C13 34888,c1(C(N(C(C)CNC(c2cccc(C(F)F)n2)=O)C)=O)nsc2c(Cl)cccc12 34889,N1(C(C2CC(NC(Cc3cc(C)sc3)=O)C2)=O)CCCCC1C 34890,Cc1ccc(C(CNC(c2occc2C)=O)NC(c2scc(C)c2C)=O)cc1 34891,O=C1CCCC(CC(=O)NCC(CC2CC2)C(=O)NC2CC(C(F)(F)F)C2)C1 34892,C1(NC(Cn2ncc(C#C)c2)=O)CN(C(=O)C(C)CC(F)F)C(C)(C)C1 34893,c1(CC)cnc(C)nc1N1CCC(CNC(=O)CN(C)CCOC)C1 34894,C1(CN(C)C(c2cc(C3CCC3)[nH]n2)=O)CN(C(c2cc(Cl)cn2C)=O)CCO1 34895,CC1CCC(C)(C(=O)NCC(=C2CN(C(C3CC4CCC3C4)=O)C2)F)CC1 34896,Cc1c(C)c(C)c(C(=O)NCC2C(C)CCN2c2ncncc2Br)c(C)c1C 34897,c1(C(=O)NCC2N(C(CCCC#C)=O)CC2)ccc(N(C)C)c(C(F)(F)F)c1 34898,c1(C(=O)NC(C(=O)NCc2ncc(C)[nH]2)C2CC2)cncc(C#N)c1 34899,Cc1ccc(CC(CO)NC(c2cnc[nH]2)=O)nc1 34900,c1(C(N2CC(CC)N(C(=O)CC3C=CS(=O)(=O)C3)CC2)=O)nccn2ccnc12 34901,C1(N(C)C(C23CSCC2C3)=O)CCN(C(=O)COc2ccccc2)CC1 34902,C1(NC(C(C)n2ccnc2)=O)CCN(C(c2ccn(O)c(=O)c2)=O)C1(C)C 34903,c1(C(N2CC(C)C(NC(c3csc(O)n3)=O)CC2)=O)cncc2c(O)nccc12 34904,C(CCC(C(=O)NCCc1cccc(C)n1)N(C)C)NC(C1C(=C)C1)=O 34905,n1(CC(=O)N(C2CCN(C(=O)C=CC(F)(F)F)C2)CCC)cnnc1O 34906,Cc1cc(CC(=O)NCCC2CCN(C(C3CCCS(=O)(=O)C3)=O)C2)ccc1O 34907,C1(CCC)CN(C(c2cc(F)ccc2F)=O)CCN1C(c1cc2n(c1)CCC2)=O 34908,C1(C(=O)NCC(C)(C2CC2)NC(c2ccnnc2)=O)CC(C)(c2ccccc2)C1 34909,C1(CCC)CCCCC1NC(c1csc(CNC(C2(CO)CCCCC2)=O)c1)=O 34910,CC1(C(N2CCCN(C(C3CCCC(F)(F)C3)=O)CC2)=O)COCC1(F)F 34911,c1(N2CC3(CN(C(c4c(C)cno4)=O)C3)C2)ccc2c(n1)CCCC2=O 34912,c1(CC(=O)NCC2CCC2NC(c2ccccn2)=O)cnc(C2CC2)[nH]1 34913,C(=O)(C1=C(Cl)CCCC1)NCC1(COC)CCCN1C(C1CC12CCC2)=O 34914,c1(C(N2CCC(COC)(NC(C3(CF)CC3)=O)C2)=O)cc(Cl)cc(C(F)(F)F)n1 34915,N1(C(C(C(C)C)F)=O)CCC(C)(NC(=O)CCc2nnc(O)nc2O)CC1 34916,c1(OC)c(Cl)ccnc1NC(C1CN(Cc2ccc(F)c(F)c2)CCS1)=O 34917,N1(C(c2cn(CCOC)nn2)=O)CCC(CO)(NC(C2CN(C)CCO2)=O)CC1 34918,C(CC(C)(C)C(=O)NCCN(S(C)(=O)=O)C)OC.N1(CC)CCN(CC)CC1 34919,N1(C(=O)NC(C)C(=O)NC2CC2)CCN(C2CCCC2)C(C)C1 34920,C1(NC(c2ccc(OC)cn2)=O)C2CC(O)C1N(C(=O)Cn1cnccc1=O)C2 34921,C1(OC)CC(C(=O)NCC(C)CNC(=O)C(C)OC(C)(C)C)N(S(C)(=O)=O)C1 34922,N1(C(C2(C)CNC(=O)C2)=O)CCCN(CCNC(=O)C=Cc2ccsc2)CC1 34923,CN1CCC(CC(N2CCCC(C(=O)NCCNC(C3(F)CC3)=O)C2)=O)CC1 34924,C(C(N=c1ccn2c(Br)cnc2[nH]1)C(C)C)NC(c1cnc2ccc(C)cn21)=O 34925,N1(C(=O)Oc2cc(C)n(C)n2)CC2CCCCC12c1ccccc1.C(C)(C)(C)O 34926,Cc1cc(F)ccc1CC(=O)NC(CNC(=O)CC1CCCC(=O)N1)CC(C)C 34927,C(C(O)C(=O)NCC(c1ccccn1)(F)F)NC(=O)CC1CCCCC1 34928,c1(N(CCN(C(c2ccc(OCCOC)cc2)=O)C)C)c[n+]([O-])ccc1[N+](=O)[O-] 34929,C1(CC(=O)NC(CCNC(c2c(C)nco2)=O)C(C)(C)C)CC2(CCCC2)CO1 34930,c1(NC(CC2C(C)C2)=O)cccc(CNC(c2cnccc2C(F)(F)F)=O)c1 34931,N1(C(CN(C)CC)=O)C2CCC1CC(O)(CNC(=O)C(C)OC)C2 34932,Cc1cc(C(=O)NC2N(C(C(=O)NCC3(C(=O)O)CCCC3)=O)CC2)cc(C)c1N 34933,N1(C(C2N(C(c3cc(SC)oc3)=O)CCCC2CO)=O)CC2(CNC(=O)N2)C1 34934,c1(C(N2C(C)CC(CNC(CC(C)C3CCCO3)=O)C2)=O)coc(S(C)(=O)=O)c1 34935,CCCCCC(C)CC(=O)NCC1(O)CCCN(C(C2(CO)COC2)=O)C1 34936,n1(CC#C)c(C)cc(C(N2CC=C(CNC(=O)Cn3nnnc3C)CC2)=O)c1C 34937,C=CC1(C(=O)NCc2ccn(C3CC(C(=O)OC)C3)n2)CCCCC1 34938,C1(NC(c2ccc(C3CC3)cn2)=O)C2CCC1N(C(=O)C(C1CCCCC1)O)C2 34939,CC(C(C)(C)CN(C)C)NC(c1cn(CCNC(c2ccn(C3CC3)n2)=O)nn1)=O 34940,CC(C(=O)N1CCN(C(=O)CN(C)CCO)C(c2ccncc2)C1)C(C)(C)C 34941,Cc1cccc(C)n1.O(NC(=O)Cn1cccn1)NC(=O)CC1CCCOC1 34942,c1(C(=O)NCCCCC(CO)NC(C(C)SCC)=O)ncc2ccccn12 34943,N1(C(C(C(=O)OC)(C)C)=O)CCC2(CC1)OCCC2NC(c1ccc(C)cc1)=O 34944,C1(C(C)NC(C2CNC(=O)C2)=O)CN(C(=O)CN2CCCCC2)CCO1 34945,c1(C(N2CC(O)(CN(C(C(C)O)=O)C)C2)=O)cn(C)nc1-c1cccs1 34946,CC(CC(=O)NCC(O)CNC(C1(F)CCCC1)=O)NC(=O)NC1CCCC1 34947,c1(C(=O)NCC(CNC(c2ccc(C(C)C)nc2)=O)(C)O)cc(CO)ccc1Cl 34948,N1(C(C(CCC)OC)=O)CCC(CO)(NC(=O)CCOc2ccc(F)cc2)CC1 34949,c1(CC)ccc(C(=O)NCC(C)N(C(=O)C(c2ccccc2C)C)C)c(C)n1 34950,N1(C(c2c(CC)occ2C)=O)CC(C(=O)NCc2csc(C)c2C)CCC1(C)C 34951,C(CNC(C1CC(=O)NC1(C)C)=O)(C(=O)N=c1cc(C)n(C(C)C)[nH]1)OC 34952,C(=O)(C1=C(C#N)CCC1)N1CCC(C(N(C)CC)=O)C1C(C)C 34953,c1(C(=O)NCCNC(c2onc(C)c2C)=O)cccc(C2CC2)c1Cl 34954,C1(C(=O)NC(C2CCN(C)C2)C)(CO)CN(C(C2CCN(S(C)(=O)=O)C2)=O)C1 34955,c1(N(C(=O)CCCC(F)(F)F)C2CCNCC2F)ncnc2n[nH]c(Br)c12 34956,Cc1cc(C(=O)NCCC2CCCN(C(=O)Cc3cnc[nH]3)CC2)cc(F)c1C 34957,C#Cc1ccc(C(N2CCCC2CNC(=O)CC(N2CCCCC2=O)C)=O)o1 34958,N1(C(C(C)C(C)(F)F)=O)CC2(CCCC2CNC(=O)C(C2CCOCC2)O)C1 34959,C1(C(N2C(CCN(C(=O)C#CC3CCC3)C)CCCC2)=O)CC2(CCC2=O)C1 34960,CCC(CC(=O)N(C)CCOCCC(N1CC=CC1C(=O)NC)=O)OC 34961,Cc1ccccc1CCC(=O)NC1(CNC(=O)C(C)C#N)CCCC1 34962,CC(C)S(=O)(=O)C(C)C(=O)NCCN(C(=O)CCCCN1CCCC1)C 34963,c1(C(=O)NCCCCNC(=O)C(c2ccccc2)F)cn(C2COC2)nn1 34964,c1(OC)cc(Cl)ncc1C(=O)NC1CC1C(=O)Nc1cc(I)ncn1 34965,CC1CC2CN(C(c3cccnc3O)=O)CC2N1C(=O)CCCC1CCCO1 34966,C1(CC(=O)NC(CNC(C(Cc2ccccc2)OC)=O)C)CCC(=O)N1C 34967,N1(C(Cc2cc(C)on2)=O)CCC(C)(CNC(=O)C(C2CCOCC2)C)C1 34968,c1(C(N2C(C3CCN(C(C(CC)=CC)=O)C3)CCCC2)=O)ccc2ccnn2c1 34969,CCC(F)(F)CC(=O)NCC1CC1NC(=O)C(c1ccnn1C)O 34970,c1(C(=O)NC2CCCC(C(=O)NC3CC3)CC2)cccn2nccc12 34971,C1(C2CC2)(C(=O)NCC(C)CNC(=O)C(=C2CCCCC2)F)CC=CC1 34972,C(=O)(C(C)(C)C(F)(F)F)N(C(c1c(Cl)ccc(OC)n1)=O)C1CC1 34973,c1(C(=O)NCCOC2CN(C(C3CC34CCCOC4)=O)C2)cn2cccnc2n1 34974,CCC(C)(CNC(c1cc(C)c(F)cn1)=O)C(=O)NOCC(O)C(C)C 34975,c1(C(=O)OC)ccc(NC(C2CCCCN2S(=O)(=O)CCCl)=O)c(Cl)c1 34976,C1(C(N)=O)(C(=O)NCC2(CCNC(=O)COC3CCC3)CC2)CC1 34977,CCC(C)CCC(O)CC(=O)NC1(C)CN(C(c2csnc2OC)=O)C1 34978,N1(C(c2c(CC)ccs2)=O)CC(CNC(c2cnnc(O)c2)=O)CC1(C)C 34979,C1(N(C(c2c(C)cc(C#N)s2)=O)C)CCCCC1S(C)(=O)=O 34980,c1(COC)ccc(C(=O)N(C(C)CNC(C2(CC#N)COC2)=O)C)o1 34981,N1(CCCCOC)CCN(C(=O)NCCCC(C)(F)F)CC1 34982,Cc1nn(C)c(C)c1C(C)C(=O)NC1CN(C(=O)C=CC2CCCC2)CC12CC2 34983,Cc1nc(=NC(=O)Nc2nn(-c3ncccc3F)cc2C)n(C)[nH]1 34984,N1(C(COCCOC)=O)CCC1CNC(c1cnsc1)=O 34985,N1(C(Cn2ccc(C)n2)=O)CCC12CN(C(c1nc(O)c(C)s1)=O)C2 34986,C(C(C)(C)CCC=C)NC(CCC=CC)(C)c1nnnn1CC(F)F 34987,C1(C(N(C(C)C)C)=O)CC2(CCN(Cc3cnc4ccccn34)CC2)C1 34988,N1(C(CC(=C)Br)=O)CC(CNC(=O)CC(CC)C2CCC2)C(C)C1 34989,C1(C(N2C(CC(=O)NCc3ccccc3F)CC2)=O)Cc2ccccc2C1 34990,O=C1CCN(C(c2ccc(N3CCOCC3)nc2)=O)c2cc(Br)ccc2N1 34991,C1(C2CCN(C(=O)CC(C)C(C)(C)C)C2)(NC(C)=O)CC1 34992,C=CC(C)(CC)C(=O)NCCC(F)(F)Cn1cc(CC(=O)OCC)nn1 34993,c1(C(=O)NC(CC=C)CNC(=O)C(C)(C)C)cc(S(N)(=O)=O)c(F)c(F)c1F 34994,c1(C(=O)NC(CCNC(CC2CCC(C#N)C2)=O)(C)C)cc(F)cc([N+](=O)[O-])c1 34995,C1(C2CCN(C(=O)COC(F)(F)F)CC2)(NC(c2c(F)ccc(C)c2)=O)CCC1 34996,Cc1nc(Cl)[nH]c(=NCC2(NC(C3CCC(C(F)(F)F)CC3)=O)COC2)c1F 34997,c1(C(C(=O)NCC)N(c2cccc([N+](=O)[O-])c2)CC)cnc2c(c1)c(C)nn2C 34998,C1(C(N2CC3C(NC(=O)Cc4ccsc4Br)(C3)C2)=O)CCCC1C1CC1 34999,Cc1[nH]nc(C(N2CCCC2C(=O)NCC2CCSCC2)=O)c1C 35000,C(=O)(CC(C)(C)OC)N(CCCNC(c1csc(-c2cn[nH]c2)n1)=O)CC 35001,C(=O)(C(O)(c1ccccc1)SC)NCC(CC)NC(=O)C(C)(C)c1ccccc1 35002,Cc1cc(=O)c(C(=O)NC2CC2CNC(c2cn(C)nc2Br)=O)cn1C 35003,CCCC(C(=O)N1CC2CN(C(=O)CCCN3CCOCC3)CC2C1)C(C)C 35004,c1(C(C)NC(=O)CNC(C2C=CC(NC3(c4cccs4)CC3)C2)=O)ccccc1 35005,C1(CNC(C(C#C)(C)C)=O)CN(C(=O)CCn2ccnc2)CC(C)(C)O1 35006,CCCC(C)CCCC(=O)Nc1cnc(Br)c(OCCC)c1 35007,C1(C(=O)NCC2COCCN2C(C2(NC(N)=O)CC2)=O)(OC)CCCOC1 35008,N1(C(=O)CC2CCC(F)(F)C2)CCC2CN(C(c3ccc(Cl)cc3Cl)=O)CC2C1 35009,c1(C(=O)NCC2(CNC(=O)CCOCC3CC3)CCC2)occ2c1CCCC2 35010,c1(CC)noc(CC)c1CC(N1CC(NC(c2conc2C)=O)CC1C)=O 35011,C1(NC(C#CC(C)C)=O)CCC2CC1CN2C(C1CCOC(=O)CC1)=O 35012,Cc1nc(C(C)C)nc(O)c1C(N1CC2(COC(CNC(C3CCO3)=O)C2)C1)=O 35013,C1(NC(C(C2CC2)SC)=O)CCCC1NC(=O)Cn1ccc(Br)n1 35014,CC(C)CC(F)(F)C(=O)N1C2CCC1CC(CNC(C1CC(C)CO1)=O)C2 35015,C#CCC(C)(C(=O)NCCC1CC1C)NC(c1cc(C#N)cs1)=O 35016,C1(C(N2C(CNC(CNC3CCCC3)=O)CC2)=O)CCc2ncnc(C)c2C1.CO 35017,CCCCCCC(C)(CC)C(=O)OC1CCOC(c2ccc(Cl)cc2)C1 35018,C(C1=CCN(C(C2CC(C)CN(C(=O)Cc3cncs3)C2)=O)CC1)OC 35019,CC1=C(C(=O)N2CC3CCC3(NC(=O)CSCc3csc(C)n3)C2)CCCO1 35020,CC1C(NC(=O)CCC2CCC(C)O2)CCCN1C(c1cn(C)c(=O)n1C)=O 35021,C(=O)(CC1c2ccccc2C(=O)N1C)NCCCCNC(CC1CC(SC)C1)=O 35022,Cc1ccc(CNC(C2CC(C)N2C(=O)CCCc2ncco2)=O)cc1 35023,S(=O)(=O)(c1ccc(=NCCS(=O)C(C)(C)C)[nH]c1)NCc1nc(C)sc1 35024,c1(C(N(CC(C)NC(=O)C=CC2CCCO2)C)=O)cc(Cl)cc(F)c1F 35025,Cc1cc(C(N2CC(C)CCC2CNC(c2cn(CO)nn2)=O)=O)c(C)nc1C 35026,C(C)(C(O)C(=O)Nc1nnc(-c2ccc(NS(C)(=O)=O)cc2)s1)OC 35027,C(=O)(C1=CC(C)CC1)NC(C)CCNC(c1ccn(C2CCC2)n1)=O 35028,C12(C(N3CCC(C)(C(=O)NC)C3)=O)COC(C1)C(NC(=O)CC(=O)NC1CC1)C2 35029,CC1CCN(C(C2(CF)CC2)=O)CC1NC(C1CCN(C2CC2)CC1)=O.C(C(F)F)O 35030,CC1CN(C(=O)CCc2cscn2)CC1NC(C1(F)CCCOC1)=O 35031,C12(COC)CC(NC(=O)CN3CCCC3C)(CN1C(=O)Cc1ccccc1C)C2 35032,C12(CC(=O)NC(CNC(C(C)(C)F)=O)C(C)(C)C)CC3CC(C1)CC(O)(C3)C2 35033,CCCC(C(=O)NOC(CO)C(C)C)NC(=O)C(F)F 35034,c1(C(N(C)CC2(NC(C3CCCCCCC3)=O)CC2)=O)c2c(nn1C)CCSC2 35035,c1(N(CCN(C(=O)C=CC2CCOC2)C)C)cc(-c2ccccc2)nc(Cl)n1 35036,c1(C(=O)NC(CN(C(C(C)SCCCC)=O)CC)C)cnc(CC(C)C)[nH]1 35037,C1(CNC(c2ccc(CN(C)C)o2)=O)CC12CCN(C(c1ccc(F)o1)=O)CC2 35038,Cc1cnc[nH]c1=NCCCC(C)NC(c1cnn(CCN(C)C)c1)=O 35039,c1(NC2C(C)CCN(C(C3CC3c3ccccc3)=O)C2)ncnc2sccc12 35040,C1(C(=O)NC(CCCCC)C)CN(C(C2(O)CCOCC2)=O)CC12CC2 35041,c1(C2C(C(=O)NCCCNC(C(C)(C)C3(C)CC3(F)F)=O)C2)ccc(F)cc1 35042,c1(C(=O)NC2CC(CNC(C3C(OC)C3C)=O)C2)occc1CN(C)C 35043,N1(C(C2C(CCC)C2)=O)CC2(C1)C(N(C(=O)C1CC1)C1CC1)CCS2(=O)=O 35044,C=CCC(C)(C)CC(=O)NC1CCCC1NC(=O)C=C(C)C1CC1 35045,CCC(CC(=O)NC(CCOCCO)C(=O)N1CC=CCC1)C1CC1 35046,c1(OC)cc(Cl)cc(N)c1C(=O)NCc1sc(N(C)C)nc1C 35047,C1(C(N(C)CC2CC(F)C2)=O)CCC(C2CC2)N1C(c1ccc(O)cc1)=O 35048,c1(-c2cn(CC(N3CCC(C#N)CC3)=O)nn2)ccc2ccccc2n1 35049,CCCCCC(O)C(=O)NCc1cc(-c2ccc(C#N)cc2)nn1C 35050,C1(CN(C(=O)Cc2sccc2C)CC)CCCCN1C(=O)CN1CCC(F)(F)C1 35051,c1(C(N2CCC(CCNC(C(C)CC(F)F)=O)C2)=O)cccc2c1CC(=O)N2C 35052,C1(OCCCNC(CC(=O)NCC#C)=O)CCN(C(=O)C(C)COC)CC1 35053,N1(C(CC2CN(C)C2)=O)CC2CC2(C(=O)N(C2CCCC(O)C2)C)C1 35054,c1(C(C)C)ccc(C(=O)Nc2cccc(NC(=O)CCC3CNC(=O)N3)c2)cn1 35055,Cc1oc(-c2ccccc2F)nc1C(=O)NCC(O)CN(C)C(c1cncs1)=O 35056,C(=O)(NNC(=O)c1ccc(CO)cc1)NC(C)CC(N)=O 35057,Cc1c(CC(=O)NC2CN(C(=O)COCC(C)C)CCC2C)sc2ccccc12 35058,N(C1CCCc2c1cnn2Cc1ccccc1)C(c1cc(C)c(O)c(C)c1)C 35059,C(=O)(C1CCSc2ccccc21)N1C(C)CCN(C(c2cnn[nH]2)=O)CC1 35060,C(C(=O)Nn1cnc2ccccc12)NC(C1CN(C(c2c(C)ccc(F)c2)=O)C1)=O 35061,C1(NC(C2CCC(NC(CCC3C(C)C3)=O)C2)=O)CC2CC1CC21CC1 35062,C(CC(C)C(=O)NCC(O)CNC(c1ccnc(NC(=O)NC2CC2)c1)=O)=CC 35063,C(=O)(CC(C(F)(F)F)N1CCOCC1)N1CCC(F)(C(N2CCOCC2)C)C1 35064,O(NC(=O)C(C)(CSC)NC(c1cnc2ccccn12)=O)C(C=C)C 35065,c1(C(=O)NCC2CC(C)OC2C)cccnc1[N+](=O)[O-] 35066,N1(C(C2C(C)C2)=O)CC2(CCC2NC(=O)CCc2cc(Cl)cc(Cl)c2)C1 35067,c1(NCC2C(NC(c3nccc(Cl)c3F)=O)CCC2)ncnc2cc(Br)sc12 35068,CCCC(C)CCCC(=O)NCC1CN(C(=O)Cc2cc(Cl)n(C)n2)CC1(C)C 35069,CC1CN(C(=O)Cc2cc[nH]c2)CC(C)CN1C(C1CC12CC(O)C2)=O 35070,Cc1cc(C=CC(N2CC(F)CC2CNC(=O)C(C)OCCC2CC2)=O)on1 35071,C(C(C)CC(C)C)NC(c1n(CCCOC)nnn1)c1ccc(I)s1 35072,c1(OC)ccc2ccccc2c1NC(C1CNCCN1Cc1cncs1)=O 35073,C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCC(CNC(C2(CC)CC2(F)F)=O)C12CC2 35074,N1(C(C(COC)OC)=O)CCN(C2CCCN(C(=O)C=C(C)C(C)C)C2)C(=O)C1 35075,C12(C(=O)NCC3CCN(C(c4cccnc4S)=O)C3)CCC(O1)c1ccccc12 35076,C1(NC(C2(CC)CCC2)=O)CN(C(=O)C(C)CSC)CCC1CO 35077,N1(C(C(C)(C)F)=O)CCC(CC(=O)Nc2ccc(-c3nn[nH]n3)cc2)C(F)(F)C1 35078,c1(CC)cc(C(=O)NC2CC2CNC(c2cncc(N)n2)=O)cc(O)n1 35079,CCC(C)C(=O)C(=O)NC1COCCC1C(=O)N(CCC(N)=O)CC 35080,N1(C(CNC(C2C(C)C2)=O)=O)CCC(C(=O)N(C2CSC2)C)(CF)C1 35081,c1(C(=O)NCC2C(N(C)C)CN(C(CC3C(CC)C3)=O)C2)c(Cl)ccnc1C 35082,S(=O)(=O)(c1c[nH]c(=NCCC2CC2(Cl)Cl)cc1C)N1CCC(OC(=O)NC)CC1 35083,C12(CC(=O)NC(CC=C)CNC(C3CCO3)=O)CC3(F)CC(F)(C1)CC(F)(C2)C3 35084,Cc1cc(C(=O)NC2(CNC(=O)CCSc3nnnn3C)CCOC2)ncn1 35085,c1(C(=O)NC2CCCC(OC)CC2)c(F)cc(Cl)cc1Cl 35086,Cc1c(CC(=O)NC2CC(CNC(C3(O)CCCC3)=O)C2)cccc1[N+](=O)[O-] 35087,c1(OC)ccc(F)cc1CC(N1CC(NC(c2cn(C)cn2)=O)C(C)C1)=O 35088,c1(Cn2cc(CCCCNC(C(C)CCN(C)C)=O)nn2)csc2ccccc12 35089,c1(C(=O)NCC2N(C(c3c(Cl)c(C)n(C)n3)=O)CC2)cncc2c1CCCC2 35090,N(C1CCOc2ccc(O)cc21)C(c1c(C)cco1)C 35091,Cc1ccc2c(c1)C(=O)N(CC(=O)NCC1COCCN1C(=O)C=C1CC1)C2=O 35092,N1(C(C2CC(C)OCC2)=O)CC=C(C(=O)N(c2cccc(C#N)c2)C)C1 35093,n1(CCOC(C)C)nc(Cc2ccccc2Br)nc1-c1cncn1C1CC1 35094,N1(C(CC(C)c2ccco2)=O)CC(CNc2ccccc2[N+](=O)[O-])OC(C)(C)C1 35095,N1(C(c2ccc(C(C)C)cc2)=O)CCCC(C)(NC(C2CCC3CC2CO3)=O)C1 35096,CCCCCCC(C)(CCC)C(=O)NC1CC(CCNC(=O)CC(C)F)C1 35097,C1(NC(Cc2nc(CC)sc2)=O)CN(C(=O)CC2C(=O)NN=C2C)C2(CCC2)C1 35098,Cc1noc(CN(C)C(=O)NCc2ccn(CC(F)(F)F)n2)n1 35099,C(CN=c1[nH]c(=NCC2CC2C(C)C)[nH]c2cccnc12)c1ccc(C)nc1 35100,C(CCCC(=O)N1CC(O)CC1C)NC(c1c(CCC)[nH]cc1)=O 35101,C1(C(=O)NC2CCN(C(C(=C(C)C3CC3)F)=O)C2C)CC(C(C)C)=NO1 35102,C1(C(N(CC(C)(C)NC(COCCCC(C)C)=O)C)=O)CCCCC1(F)F 35103,N1(C2CCN(C(C3C(C)C3)=O)CC2)CCC(NC(=O)C=CC(=O)NC2CC2)CC1 35104,N1(C(C=CC=CCC)=O)CCC(O)C(NC(=O)CC2CCN(C)C2)C1 35105,c1(OC)nccc(C(N2CC(NC(c3nc(C)ncc3Br)=O)C(F)C2)=O)c1F 35106,CC1(C)OC2(CN=c3ccc(C(F)(F)F)c[nH]3)CC1(C(=O)Nc1cnco1)C2 35107,N1(C(CC)C(N)=O)CCC(NC(c2c[nH]nc2C)=O)C(O)C1 35108,C(=O)(CC(C)C(=O)OC)NCC1(F)CCC(NC(c2cc(CC)ncc2)=O)C1 35109,c1(NC(c2c(C(C)C)nns2)=O)ccccc1I 35110,c1(NC(C2OCCN(C(c3c(OC)ccnc3)=O)C2)=O)cc(Cl)nnc1OC 35111,C1(C(=O)NC(CC)CNC(c2ccc(C)cn2)=O)CC(O)CN1C(=O)N(C)C 35112,C1(C)(C(N(CC#C)CC=C)=O)CCCN1C(=O)CCn1cc(C(=O)OC)cn1 35113,c1(C(=O)NC2C3CN(C(c4ccc(C(C)=O)cc4)=O)CC32)c(F)cc(F)cc1Cl 35114,N1(C(C(CSC)(C)C)=O)CCC(CNC(C2CCCC(CF)C2)=O)C(O)C1 35115,c1(C(N(CC(CNC(C(C)SCCCC)=O)C)C)=O)ccc(-n2ccnn2)cc1 35116,c1(C(N2C(CC(=O)NCC(C)C3CC3)C3CCCC32)=O)cc2ccccc2o1 35117,CC1CCC=C1C(=O)N1CCN(C)CC1CNC(=O)CN1CCOCC1=O 35118,c1(SC)cccc(NC(C2CCC(NC(=O)CC(=O)OC(C)C)CC2)=O)c1O 35119,O=C(O)CCC(F)(F)C(=O)N1CC2CC1CN2Cc1ccc(F)cc1 35120,c1(SCCN(C(=O)C(C(=O)OC)OC)C)cc(Cl)cc(Cl)c1 35121,N1(C(CCOCCC)=O)CCCC2CN(C(c3cncc(NCC)c3)=O)CCC12 35122,C=CCC(C)C(=O)N(C1CCCN(C(=O)C=C(C)CCC)C1)CCO 35123,c1(OC)cc(C(=O)NC(C)CC(C)NC(c2cnn(CCO)c2)=O)ccc1Cl 35124,C1(C(N2CCC(O)(CC)C2)=O)COCCN(C(=O)COCC(=O)NC)C1 35125,C1(C(=O)NC2(C)CCN(C(C(CSC)O)=O)CC2)Cc2ccccc2S1 35126,C1(CN(C(C(C2CCCC2)NC(C(C)=C(C)C)=O)=O)C)C(C)(C)C1(C)C 35127,CCCCC(F)C(=O)NCC1COC(CNC(=O)Cc2csc(C3CC3)n2)C1 35128,C(=O)(C(F)(F)C(C)O)NC(C)CCCNC(c1cc(F)cc(Cl)c1)=O 35129,c1(OC)ccc(-n2nc(-c3cccc(Cl)n3)nc2C2CCOC(C3CC3)C2)cn1 35130,C=C=C(C)CC(=O)NC1(CC=C)CCN(C(c2cnn(C(C)CC)c2C)=O)C1 35131,C(CC(C)(C)C(=O)NCC(N1CCOCC1)=O)NC(C=CC=CC)=O 35132,c1(NC(C2C3CN(C(CCCC(C)C)=O)CC32)=O)cc(Cl)c(Cl)cc1C#N 35133,N1(C(c2cnn(C3CC3)c2)C(=O)NCC2CCCO2)CC2CC(O)C(O)CC2C1 35134,c1(OC)ccc(C(=O)NCCCN(C)C(c2c(F)cncc2Cl)=O)c(O)c1 35135,C1(C(=O)NCCCC2CCCN2C(=O)CN2CCSCC2)CCCCCC1(F)F 35136,N1(C(C2CC(C)SCC2)=O)CCN(C(=O)Cn2cccc2)CC1CO 35137,c1(NCc2cccc(OCCOC)c2)[nH]c(=NCC2CC2C)nc2ncn(C)c12 35138,c1(OC)c(C(=O)NCC(C)CN(C)C(c2cnc(C)nc2C)=O)cccc1Br 35139,C(C)(CC(=O)NC1(CCC(=O)NCC(O)CCC2CC2)CCCC1)=C(C)C 35140,Cn1cncc1CCNCC1(C)CCN1C(=O)COC(=O)CO 35141,C1(NC(C=C(C)C(C)C)=O)CCN(C(=O)C(C)SC(F)(F)F)C1C1CC1 35142,N1(C(CCN(C(C)=O)C)=O)CCC(CN(C(=O)C(F)(F)c2cnccn2)C)CC1 35143,CN1N=CC(CC(=O)N(CC(CO)(CO)NC(=O)CC2CCCC(C)C2)C)C1=O 35144,CCC(CC)CCCC(=O)N1CCC2CN(C(c3nn(C)cc3Cl)=O)C2C1 35145,N1(C(C(C)C(F)F)=O)CCC(C)(NC(c2cc(C3CC3)cc(F)c2)=O)CC1 35146,Cc1ccc(CCCC(=O)NC2CCCC2CNC(=O)Cc2cn(C)nn2)s1 35147,C1(C)(CNC(CNS(CCOC(C)C)(=O)=O)=O)CCCN1C(=O)CSC(F)F 35148,N1(C(c2c(C)noc2)=O)CCN(C(=O)CCn2cccn2)CC1CO 35149,C(=O)(C1=CS(=O)(=O)CCC1)NCC1CC(NC(C2C(C)OCCC2)=O)C1 35150,CCC(C)CC(C)C(=O)N1CCC(F)(CNC(=O)CC2(CO)CC2)CC1 35151,c1(CC(=O)Nc2ccc3c(c2)OCC3)noc2ccc(Cl)cc12 35152,N1(C(C=CCOCCOC)=O)CCCC1(C)CNC(=O)CCC1CCC(=O)N1 35153,C1(CNC(C(N2CC(C)C2)C)=O)(CNC(C2(C)CCSCC2)=O)CC12CCC2 35154,c1(C(=O)NCC2(OC)CN(C(c3cc(C)ncc3C)=O)C2)ccn(O)c(=O)c1 35155,C1(C)(C(=O)NC2CCC(NC(c3ccc(CC)[nH]3)=O)C2)CCC(C)(C)CC1 35156,C(=O)(C(CO)C(C)(C)C)NCc1c(C(=O)NCC(C(=O)NC)(C)C)occ1 35157,C1(NC(c2c(C(C)C)n[nH]c2)=O)CCCN(C(=O)C(C2CCC(=O)N2)C)CC1 35158,c1(C(=O)OC)cc(F)c(Br)c(S(=O)(=O)NC(=O)COc2ccc(C)cn2)c1 35159,O=C(CCCNC(c1cccnc1)=O)NCC1CN(C(c2cc(Cl)c[nH]2)=O)C1 35160,c1(CN(C)C)c[nH]c(C(=O)NC2CC2NC(=O)COCC2CCCO2)c1 35161,N1(C(C2(COC(C)C)CC2)=O)CC(C2CCCCN(C(C3COCCO3)=O)C2)C1 35162,c1(C(=O)NCCC2CC(NC(c3cn(CCC)nc3C)=O)C2)nnc(O)cc1O 35163,N1(Cc2c(C)cccc2)CC2(CN(C(c3ccc(Br)cc3CO)=O)CCO2)C1 35164,C(=O)(CCCCC(=O)NC1CN(C(=O)CSc2nnnn2C)CC(C)(C)C1)NC 35165,N1(C(COCCNC(C(C2CCCCC2)C)=O)=O)CCC2(CC(F)C2)C1 35166,N1(C(Cn2c(C)ccn2)=O)CCC(O)(CN(C)C(C2(C)CCCC2C)=O)CC1 35167,CC(C)CCCOCC(=O)NCC(C)N(C(=O)CC1CCN(C)C1)C 35168,N1(C(C(C)(C)NC(=O)NCC)=O)CC(NC(c2nnccc2C)=O)C(C)(C)C1 35169,C12(COC)CC(CNC(C3CCCO3)=O)(CN1C(c1nonc1N)=O)C2 35170,O=C(CCCC(F)(F)F)NC1CC(O)CN(C(=O)COC2CCOC2)C1 35171,c1(OCC)oc2ccccc2c1C(=O)NCC(CC)NC(C1CC2CC1CO2)=O 35172,c1(OC)ccc2cccnc2c1CNc1cc(N2CCCS2(=O)=O)ccc1F 35173,c1(C(C(=O)NCCC#N)N(CC)CC2CCCO2)nc2c(s1)CC(C)CC2 35174,CCCCCCC(C)C(=O)NC(C(=O)NC1CC(F)(F)C1(C)C)C(C)C 35175,C12(C(N(CCC(=O)NC(CC=C)C3CC3)C)=O)COCC1C2 35176,N12CCCCC1C2=O.c1(SCCn2cc(C(C(C)(C)C)O)nn2)ccnc(SC2COCC2)c1 35177,C1(CNC(C2C(COC)CC2)=O)COCC1NC(=O)COc1cccnc1 35178,CN=c1ccc(CNC(=O)CC2CCN(C(=O)CC3CCN(C)C3=O)CC2)c[nH]1 35179,c1(OC)cc(C2(C(N3CCCC(C)(NC(=O)CCC(N)=O)C3)=O)CC2)ccc1C 35180,C(N=c1nc2sccc2c(N2CCC(C)(C(N)=O)C2)[nH]1)c1[nH]n(C)c(=N)n1 35181,N1(C(=O)CC2CCCC2)CC(C2CCCN(C(=O)C(c3cccc(Cl)c3)O)C2)C1 35182,c1(C(=O)NCC(CCC)CCO)ccc(Br)cc1N=[N+]=[N-] 35183,c1(NC(N2CCOC(C3CCC3)C2)=O)cc(F)c(CO)c(F)c1 35184,C1(F)(C(=O)OC)CN(C(=O)CONC(c2cccnc2)=O)C1 35185,N1(C(C(CC)OCC)=O)CC(N=c2nc(C(C)(C)C)[nH]s2)CC(C)(C)C1 35186,N1(C(c2c(C)nsc2)=O)CCCC2(NC(=O)CSC(C)(C)C)CCCC12 35187,N1(C(C2CCN(CC#C)CC2)=O)CC=C(CNC(c2nncn2C)=O)CC1 35188,N1(C(CSCC=C)=O)CC2CCC(C1CO)N2C(c1ccc2c(n1)CCCC2)=O 35189,c1(C(N2CCC(NC(C(C)OCCCC)=O)C2)=O)ncccc1C(F)F 35190,[N-]=[N+]=NCC(C(=O)NC1(C2CC2)CC1)NC(=O)CCC1CCCC1 35191,C12(NC(=O)COC3CCCC3)CCN(C(c3cccc(O)c3Cl)=O)CC1C2 35192,C#CCCC(C(=O)NCC(C)C#N)NC(=O)CCCCCN(C)C 35193,n1(CC)nnc(C)c1C(=O)NC(C)C(C)NC(c1cnn(C)c1C(F)F)=O 35194,C1(NC(CC(C(C)C)C)=O)CCCC12CCN(C(=O)C(C)CS(C)(=O)=O)CC2 35195,c1(OCC)ccc(Br)c(-c2nnc(CCC(N3CC(=O)NCC3C(C)C)=O)o2)c1 35196,O=S(=O)(c1cccc(F)c1F)N1CCC(OCc2ccccc2)C1 35197,c1(C(=O)OCc2cn(CC(C(=O)NC3C(C)CCC3)O)nn2)c[nH]nc1[N+](=O)[O-] 35198,N1(C(c2cnc(COC)s2)=O)CCN(C(=O)CC2CN(C)C2)C(C)CC1C 35199,N1(C(COCCC=C)=O)CC2(CC2)CC1CN(C(=O)CSCCC(F)(F)F)CC 35200,C(=O)(C(C)(C)CCOC)NC1CCCC(CF)C1.C=C1CC2(C1)C(=O)NC2 35201,Cn1ccc(C(N2CC(C(=O)NCC=CCl)CC2(C)C)=O)cc1=O 35202,C1(C(=O)NCC2CCN(C(CC3C(C)(C)C3)=O)CC2)CCOC2(CCOCC2)C1 35203,CC1(C)CC(O)(C(=O)NCC(C2CCCC2)NC(=O)CC2CCCOC2)C1 35204,C1(C(=O)NC2CC(C)(CNC(c3cc(CC)[nH]n3)=O)C2)(OC)CCC(C)C1 35205,Cc1cc(F)c(C(N2CC3CN(C(=O)C(n4ccnc4C)C)CC23)=O)c(F)c1 35206,Cn1nc(C(=O)NC2CCCC2NC(C2CCC3CC23)=O)c2c1CCC(C)(C)C2 35207,N1(C(C(CC)C)=O)CC2CCC(C(=O)NCCc3ncn(C)n3)(C2)C1 35208,Cc1nccc(C(=O)NC2(CNC(C34CC5CC3C4C5)=O)CCOC2)c1O 35209,N1(C(Cc2ccc(C)o2)=O)C2CCC1CC(CC(C)NC(=O)C(C)CCO)C2 35210,c1(CC(=O)NC2CN(C(CC(c3c(C)n[nH]c3C)C)=O)C2)c(F)cccc1Cl 35211,S(C1CCc2c(F)cc(F)cc21)C(=O)Nc1cccc(C)c1 35212,C1(OC)CC2(CCC(C(N3CC4CCN(C(=O)O)CC34)=O)CC2)C1.C(C)(C)(C)NC=O 35213,C(CC(CC)C(=O)NCCN(CCCN(C)C)C(c1cc(F)n[nH]1)=O)=CC 35214,CCCCCC(C)CC(=O)N(C(CNC(=O)CN1C(=O)C(C)C(C)C1=O)CC)C 35215,CCC(C)C(O)C(C)C(=O)N1CCC(NC(C2CCC3CC23)=O)C1 35216,CCC(C)(C)C(C)CC(=O)NC1(CNC(=O)C=Cc2cc(Cl)ccc2Cl)CCC1 35217,C1(CNC(C2CCC(CC)O2)=O)CC(NC(c2cnc[nH]2)=O)CC1O 35218,N1(C(=O)CN2CCCC2)CC2CN(C(c3cccc4cc[nH]c34)=O)CC2C1 35219,N1(C(CC(COC)C)=O)CCCCC(CNC(=O)C=C2CCC(C)(C)CC2)C1 35220,N1(C(c2c(C)cccc2F)=O)CC(NC(=O)Cc2ccon2)CC2(CC2)C1 35221,CCCCCCC(F)C(=O)NCC12COC(CNC(=O)CC(C)(C)O)(C1)C2 35222,c1(C(=O)NCC2N(C)CCN(C(=O)C=C3CC3)C2)cnn2ccn(C)c12 35223,C=CCCCCC(=O)N1CCC(OCC(=O)NC(CCF)C(=O)OC)C1 35224,C=CCC(CC)C(=O)NC1CCCCC1C(N1CC(O)(COC)C1)=O 35225,c1(NCC#CCC)cc(C2(C#N)CCC2)ccc1OC 35226,Cn1nccc1C(=O)NCCC(O)CNC(c1c[nH]c(Br)c1)=O 35227,CC1CCN(CCC(=O)NCCCCCCNc2ccnc(OCCO)c2)CC1 35228,CCC(CCCC(=O)N1CCCCC1C)NC(=O)C(C)(C)c1ccno1 35229,Cc1nn(C)c(C)c1Cn1cc(CCN(C)CCO)nn1.c1(N)nccc(OC)c1F 35230,N(C(=S)N1CC(CO)CC(C)C1)c1ccc(OC)c(Cl)c1 35231,CC(C)CC(CNC(=O)C1=CCCCO1)C(=O)NC(C1(O)CCCC1)(C)C 35232,S(=O)(=O)(c1cc(C(=O)NCCNC(c2cnsn2)=O)co1)NC(C)(C)C 35233,c1(-c2nn[nH]n2)ccc(CNCC2CC(C(=O)OCC)C2)c(C)c1 35234,C1(C(=O)NCC2N(C(C(C(=O)OCC)(C)CC)=O)CC2)CCc2ncnc(C)c2C1 35235,C(C1=NOC2COCC12)SCC(C(=O)N1CCC1)NC(=O)CCCn1cccc1 35236,CC1CCC(CO)N(C(=O)NN2CCC(c3ncc[nH]3)CC2)C1 35237,Cc1cccc(-c2cccc(C(=O)NCC3CC(C)N(C(=O)C=C(Cl)Cl)C3)c2)c1 35238,c1(C(=O)OC)cc(C(=O)NCCCOCCNC(c2cnnc(O)c2)=O)n(C)n1 35239,C12(C(=O)NC3CN(C(COCc4onc(C)n4)=O)C(C)C3)CCCN(CC1)C2 35240,c1(C(N2CC3(CCN3C(C3(F)CCCCC3)=O)C2)=O)ccc(Cl)c(F)c1F 35241,c1(NC(N2CCC(Nc3nnnn3CCC(F)(F)F)C2)=O)ccc(Br)cc1 35242,C1(CC(NCP(OCC)(C)=O)=O)CN(C(c2ccnc(COC)c2)=O)CC12CC2 35243,N1(C(CCc2cc(C)ncc2)=O)CC2CN(Cc3ccc(Cl)cc3F)C2C1 35244,N1(C(C(CO)N(C)C)=O)CCC2(C1)CN(C(=O)CS(=O)(=O)C(C)(C)C)CCO2 35245,N1(C(c2ccn(C)n2)=O)CC2CC1C2NC(c1cccc(-n2cncn2)n1)=O 35246,c1(OCC)cc(C(N2CCC(CCNC(=O)Cc3cc(C)ns3)C2)=O)[nH]n1 35247,N1(Cc2c(OC)cco2)CCCC(NC(c2cnc(Cl)cc2I)=O)CC1 35248,C(=O)(C(C)(C)CC(F)F)NCc1c(C(=O)NCC(C#C)OC)con1 35249,c1(CN(C(=O)Nc2ccccn2)CC2CCN(C(=O)C(F)(F)F)C2)ccccn1 35250,C(=O)(C(O)C(F)(F)F)N1CCC(CCC2N(C(C=CC)=O)CCC2)CC1 35251,c1(N2CC(C3N(C(C(C(C)C)F)=O)CCCC3)C2)ncnc2cccc([N+](=O)[O-])c12 35252,c1(C(N2C(CNC(CSCC)=O)CC(C)CC2)=O)n[nH]c2cc(C)ccc12 35253,N1(C(C2(COC)CCC2)=O)CC2CCC1C2NC(=O)CCc1ccc(Cl)cc1 35254,C1(C(N(CC)Cc2occc2C)=O)CN(C(c2ccnn2C2CC2)=O)C(C)(C)C1 35255,C1(NC(C(C)c2cncs2)=O)CN(C(c2cnc(N)c(N)c2)=O)CC12CCC2 35256,C(C1OCc2ccccc21)N(C1CC(n2nnnc2C(F)(F)F)C1)CC 35257,C1(NC(CCCCNC(C)=O)=O)CC2(C1)CN(C(=O)CC1C(C(C)=O)C1(C)C)C2 35258,c1(OC)ccc(C)nc1C(=O)NC1CC1CNC(c1ccc(C(C)C)cc1C)=O 35259,C1(NC(C2C(C)CCS2)=O)CCC(NC(=O)C(C)(C)c2ccc(Cl)s2)CC1 35260,c1(C(=O)NCC2CCCN(Cc3c(O)cccc3O)C2)cccc2sccc12 35261,N1(C(c2c(CC)[nH]cc2)=O)CCCC(NC(c2csc(S(N)(=O)=O)c2)=O)C(F)C1 35262,N1(C(C(C(CC)C)O)=O)CCCC2(C1)CN(C(=O)CCc1nc(O)n[nH]1)CCO2 35263,c1(CNC(=O)CNC(=O)CNC(C)=O)cc[nH]c1C(=O)NCC1(OC)CCCC1 35264,C(c1cccc(O)c1)=CC(N1C2CN(C(c3cccnc3C(F)(F)F)=O)CC21)=O 35265,c1(CC(N2CCCC2Cn2cc(CCN3CCCC3CO)nn2)=O)sccc1Cl 35266,N1(C(C(c2ccc(Cl)s2)C)=O)CCC(NC(=O)Cc2ccc(O)c(Cl)c2)CC1C 35267,Cc1cc(C)n(C(C)C(=O)NCCC2COCCN2C(=O)CC2CCCCC2)n1 35268,c1(CCN=C(NCCOC(CC)C)NCC2CC(F)(F)C2)ccc(S(N)(=O)=O)cc1 35269,c1(C(N2CC3(CN(C(c4ccc(C)s4)=O)C3)C2)=O)cc(N)cc(C)c1F 35270,c1(NCc2ccc(Oc3ccc(Br)cc3)nc2)cccc2ncsc12 35271,CCC(C(=O)NCC1CC(C)CN(C(=O)C(n2nccc2C)C)C1)C(F)(F)F 35272,CN1CCN(C(=O)COC2CN(C(=O)C(F)C(C)(F)F)C2)CC12CCC2 35273,N12CCC3(CC(=NO3)C(=O)NCc3cc(Cl)cc(OC)c31)C2.c1(OC)nnco1 35274,C1(C(N(C(CO)C2CC2)C)=O)CC12CCN(C(=O)CCC1CC1)C2 35275,c1(C(C)(C)C)nnc(N(CCCNC(C2CN(C3CCOCC3)C2)=O)CC2CC2)s1 35276,C(=O)(C(CC(N)=O)SC)NC(C1(OC)CCN(C(c2ccc(C(F)F)o2)=O)C1)C 35277,c1(OC)ccc(C(N2CCC(CCNC(C)=O)CC2)C(=O)NC2CCC2)c(Cl)c1 35278,C(N=c1cc(C(F)(F)F)nc[nH]1)C1(CCNCC=C(C)C(C)(C)C)CC1 35279,C(=O)(CCCCN(C1CCCC1CNC(C1CC(OC)C1)=O)C)NC 35280,CCCC(C(O)C(=O)N1CCc2c[nH]nc2C1)NC(=O)C=CC(F)(F)F 35281,N1(C(c2nc(C(C)C)sc2)=O)CC(NC(C2(C(F)(F)F)CC2)=O)CC1C 35282,N1(C(C(CC)C#N)=O)CC(O)(C2CCN(C(=O)Cc3cn4ccsc4n3)CC2)C1 35283,CC(C)(C(=O)NCC1CC(NC(=O)Cc2ccno2)C1)C(F)(F)F 35284,N1(C(CN2CCC(=O)CC2)=O)CCOCC(NC(c2ccn(CCF)n2)=O)C1 35285,c1(C(=O)NCCOCCCNC(C2C(C)CCS2)=O)cc2sccc2s1 35286,C(C)(C)(CCCC(=O)NC(C(C)C)C1CC1)NC(c1ccc(OC)cc1)=O 35287,c1(NC(C2C3CN(C(C4CCC(C)CO4)=O)CC32)=O)nc2cc(F)ccc2s1 35288,C1(CC)CCCCCCN1C(C1CCOCCN1C(C1CCSCC1)=O)=O 35289,N1(C(c2cncc(C(C)=O)c2)=O)CC2CC(C1)N(C(=O)CC1CC=CCC1)C2 35290,C1(C(=O)NC(c2nocc2C(=O)NC(c2cccc(F)c2)C)C)CCCCC1O 35291,C12(CNC(C3(C)COCCO3)=O)CCC1CN(C(c1cc3occc3[nH]1)=O)C2 35292,C12(NC(c3cc(CCC)on3)=O)CCC(C1)N(C(=O)CCCCN(C)C(C)=O)C2 35293,c1(NCCC(=O)NCC(C)N(C(C(C)NC(=O)OC)=O)C)ccccn1 35294,C(CC(=O)NCC1CN(C(c2nc(Br)c[nH]2)=O)C1)(C(F)(F)F)OC 35295,Cc1cc(CNCC(=O)NC(c2ccc(Cl)cc2)C)c(C)nn1 35296,C1(C(=O)NCC2(C(C)C)CC2)C2CC3C(C2NC(C2(C(N)=O)CC2)=O)C13 35297,N1(CC(=O)NC(C)CN(C(=O)CCc2cscc2Br)C)CCCCCC1 35298,N1(C(c2c(C)nc(CC)s2)=O)CCC(NC(=O)CCN(CC)CC)C(CO)CC1 35299,c1(CC(=O)NC(C(C)C)CCN(C)C(C2CC(C)(C)C2)=O)ccccc1[N+](=O)[O-] 35300,Cc1cc(Br)ccc1CCNC(C1CC2CC2N1C(=O)CNC(=O)CC(C)C)=O 35301,c1(N(C)CC)ccc(C(N2CC(n3cc(C(C)(O)CCO)nn3)C(C)C2)=O)cc1 35302,c1(NC(C2CC(F)CN2C(=O)Cc2c(F)cccc2F)=O)cccc2c1OCO2 35303,c1(C(=O)NC(CC(C)NC(C2CC(CC)C2)=O)C)ccnc(C(F)F)c1 35304,c1(OC)cc(C(=O)N(CC(C)N(C(=O)CN2CCCC2C)C)C)[nH]n1 35305,c1(NC2C(C)SCC2)ccc(S(=O)(=O)NCC(C)(C)CO)c(Br)c1 35306,C12(NC(C3CC(OC)C3)=O)CN(C(=O)COC(C)=O)CC1CS(=O)(=O)C2 35307,C1(C(=O)NCC23OCC(NC(C4(C)CC4)=O)C(C2)C3)COc2cc(Cl)ccc2C1 35308,CC1CNc2c(C(=O)NCCN(C)C(C3CCC(N=[N+]=[N-])CC3)=O)cnn2C1 35309,C1(N(C2CCOC2C)C(c2cccc(OC(C)=O)c2)=O)CCNCC12CC2 35310,C(C1CN(C(=O)CCN(C)C2CC2)CC1C(=O)N(c1ccncc1)C)=CC 35311,O=c1c(-c2nc(CCO)nn2CCc2cnc[nH]2)c[nH]cc1F 35312,N1(c2c(C(C)=O)cccn2)CCC(NC(=O)C(C)n2cnnn2)C(O)C1 35313,Cn1nc(C(=O)NCC2(C(=O)NCC3CCCNC3=O)CCCO2)cc1Cl 35314,c1(C(C)(C)C)cc(C(=O)NCC(O)CNC(=O)CCOCC(F)(F)F)cs1 35315,C1(CC#C)(C(=O)N(C)CC2CCOCC2)CCN(C(=O)CCc2conc2C)C1 35316,N1(C(C(CC)F)=O)CC2CCOC2(CNC(c2cc(OC(C)C)ccc2Cl)=O)C1 35317,N1(C(c2c(CC)ncs2)=O)C(CNC(c2cc(CC(C)C)on2)=O)CC2CC12 35318,C(=O)(C1CCCc2cn(C(C)C)nc21)NCC1N(C(c2c(C)nns2)=O)CCC1 35319,c1(OC)ccc(C(C)=CC(=O)NC2CCC2NC(c2csc(CO)n2)=O)cc1 35320,CC(C)C(C(=O)NC1CN(C)CCN(C)C1)C(C)NC(C1CCCCC1O)=O 35321,c1(CC(=O)NC2CCCCN(C(C(CCCC)=O)=O)C2)csc2cccc(F)c12 35322,C1(NC(CCC(=O)NC)=O)(CNC(c2cccnc2F)=O)CCCCC1C 35323,N1(C(C2CCCSC2)=O)CCCCC2(CCN(C(=O)C(C3CCOCC3)O)C2)C1 35324,c1(C(=O)NC2C(CNC(=O)Cn3cnnc3O)C2)cc2ccc(Cl)c(F)c2[nH]1 35325,c1(C(=O)NCCC2CCC(NC(c3c(CC)occ3)=O)C2)ccc(Cl)cc1NC 35326,Cc1ccc(S(=O)(=O)N(C(Cn2ccnn2)C(=O)N(C)C)C)cc1C 35327,C1(CNC(c2cnn(C)n2)=O)C(C2CC2)CCN1c1ncnc(Cl)c1F 35328,CC1(C)C(CNC(C2CCCCCC2)=O)CCN1C(C1C(C)(C)C1(F)F)=O 35329,C(C(C(=O)NCC1(CNC(C2CC(C(=O)OC)C2)=O)CC1)N(C)C)OC 35330,N1(C(CN(C(COC)=O)C)=O)CC2CC2C1C(=O)NC(CO)CCOC 35331,Cc1ccc(N)cc1S(=O)(=O)NC(c1ccc(OC(C)(C)C)nc1)=O 35332,c1(C(=O)NCC2(O)CN(C(C3(C(C)C)CNC(=O)C3)=O)C2)nn(C)c(Cl)c1Cl 35333,c1(NCC2CN(C(c3[nH]cc(CC(C)C)c3)=O)CC2C)ncnc2c1nnn2C 35334,CON(C(=O)CC1=CCOCC1)C(C)NC(c1ccc(C)nc1)=O 35335,N1(C(CC2CC(=C)C2)=O)CC2CCN(C(c3cc(N)cc(OC)c3OC)=O)C2C1 35336,c1(C(N(CC(CC)NC(C2(c3cccs3)CC2)=O)C)=O)cnc(O)n(C)c1=O 35337,O=C(C1=CCCSC1)NC1CCN(C(=O)C=Cc2ccccc2)C1 35338,C12(C(=O)NCC3C(C(=O)OCC)CCO3)CC3CC(C1)CC(F)(C3)C2 35339,Cc1c(C(=O)N(C)CCC2CCCCN2C(=O)C#CC2CC2)cccc1CO 35340,c1(C(=O)NC(CCCC)CNC(c2ccco2)=O)cccc(OC)c1OC 35341,C(CC(=O)NCC1(NC(=O)CN(C2CCCC2)C)CC1)N(C)CC 35342,c1(C(=O)NCCC(=C)CNC(c2cc(Br)c(C)o2)=O)cccc(CC)n1 35343,c1(OC)cc(C(=O)NCCC(C)(C)NC(=O)CC2CNC(=O)C2)cnc1Br 35344,C12(NC(c3c(C)cncc3)=O)CC(CNC(C3C=CCC3)=O)(C1)OC2C 35345,C(=O)(C1=NOC2COCC12)N1C(C)CN(C(C(C)=NOCC#N)=O)C(C)C1 35346,Cc1ccc(NNC(=O)Cn2cc(C3CCC(C#N)C3)nn2)cn1 35347,N1(C(c2ccc(NC(C)=O)nc2)=O)C2CCC1CN(C(=O)COC1(C)CCC1)C2 35348,c1(C(N2C(CN(C(=O)COCC3CC3)C)CCC2)=O)ccc(F)c2ccncc12 35349,C=CC(C)(O)CC(=O)NC1C2CC(NC(=O)Cc3nc[nH]n3)CC12 35350,C1(CCOC)CCCCN1C(=O)C(N1CCC(Cn2cnnc2)CC1)=O 35351,c1(C(=O)NC(CNC(C2(C)CCC(C)C2)=O)C)cnn2ccccc12 35352,C1(C(N(CCO)CC)=O)CC12CCN(C(=O)Cn1ccnc1C)C2 35353,c1(C(N2CCCC(CN(c3ncncc3Br)C)C2)=O)cncc2c1CCCC2 35354,N1(CC(c2ccc(F)cc2)NC(=O)Nc2ccc(I)cc2)CCCS1(=O)=O 35355,CC1(F)CCC(C(=O)NC2CCCC2NC(c2ccc([N+](=O)[O-])o2)=O)CC1 35356,CC1(C)CCC(CO)N(C(=O)C(c2cc(F)c(F)c(F)c2)O)C1 35357,c1(C(=O)NCC2N(C(C(C)NS(CC)(=O)=O)=O)CC(O)C2)cccc(F)c1C 35358,CC(C)(C)C(O)C(=O)NCC1CN(C(c2ccnc(C(F)(F)F)n2)=O)CC1(C)C 35359,Cn1nc(C(=O)NC2CCC(NC(c3coc(CC4CC4)n3)=O)C2)cc1C#N 35360,N1(C(C2(CC)CC2)=O)Cc2cccc(CNC(=O)Cc3cn[nH]c3)c2C1 35361,c1(OC)ccc(S(=O)(=O)OCC(=O)Nc2cc(Cl)cs2)cc1[N+](=O)[O-] 35362,N#Cc1ccc(C=CC(=O)NC2CC2CNC(c2cn(CC3CC3)cn2)=O)cc1 35363,CC(C1Cc2ccccc21)NC(C1C(C)(C)C1(C)C)=O 35364,Cc1nc2cc(C(=O)NC3C4CN(C(=O)C(O)C5CC5)CC34)ccc2n(C)c1=O 35365,CSC1=C(C(=O)NCC(C2CC2)N(C(=O)C(CO)c2ccccc2)C)CCCC1 35366,C1(C(=O)N(C)CCOCCN(C)C(c2c[nH]cc2C2CC2)=O)(CC)CC1(F)F 35367,C1(NC(=O)NCC(C)OC)CCN(C)C2(CC2)C1 35368,C1(NC(C(CC)N(CC)CC)=O)CCN(C(=O)C=Cc2ccsc2)C1C 35369,c1(SC)c(C(=O)NCC2(CNC(c3cnn(C)c3Cl)=O)CC23CCC3)cnn1C 35370,c1(C(N2CC(C(C(=O)N(C)Cc3csc(C)c3)OC)C2)=O)cc(CO)n[nH]1 35371,C1(OCCN(C)C(=O)NCC2COC2)C2CCC(C2)N1C(=O)OC(C)(C)C 35372,C12(C(=O)NCC(C)(C)CNC(C3(CO)CC3(F)F)=O)CC=CC(C1)OC2 35373,C=Cn1nccc1C(N1CCSCC1C(=O)N(C(CC)C1CC1)C)=O 35374,c1(C2C(C(N3C(C(=O)NCCC(=O)O)CC3)=O)C2)ccccc1OC(F)(F)F 35375,Cc1ncncc1C(=O)NCCn1cc(CNC(C2CC2C(C)(C)C)=O)nn1 35376,N1(CCNC(c2c(C)occ2)=O)CCC(NC(c2c[nH]c(=S)cn2)=O)CC1 35377,C1(NC(CS(CC)=O)=O)CCCCCC1C(N1CCN(C)C(C)C1)=O 35378,CC1CC(C(=O)NC2C3CCC2N(C(=O)Cc2ccon2)C3)=NO1 35379,C(CCN(C)C)(C(=O)NCCOC1CC1)NC(C1(COC)CCCO1)=O 35380,C1(NC(C=CC(=O)OCC)=O)C2CC(O)C1N(C(=O)Cc1csc(NC=O)n1)C2 35381,CC1(CNC(=O)C=Cc2ccco2)CN(C(=O)CCN2CCC(F)C2)CCO1 35382,C(=O)(C#CC(C)(C)CNC(C1(C)CC1(C)C)=O)NC1C(C)COC1 35383,CCCN=c1[nH]c2c(c(=NC(C)c3ccc(Cl)nc3)[nH]1)CSC2 35384,c1(C(=O)NC2C(N(C)C(c3ccnnc3O)=O)CCCC2)ccc([N+](=O)[O-])o1 35385,N1(C(c2nc(C)oc2C)=O)CCN(C(c2cc(=O)c(O)c[nH]2)=O)CC(O)C1 35386,N1(C(C=CC)=O)CCC2(CC1)CC(NC(=O)C(C)Sc1nnnn1C1CC1)CO2 35387,CCC(C)(CCNC(=O)C(F)C1CCCC1)NC(c1ccsc1OC)=O 35388,C(=O)(C(C(C(C)C)OC)N1CC(O)CC1CNCC(F)F)NC(C(=O)OC)C 35389,C(C(C)(CO)CO)N(C(=O)CN(C(=O)C(CO)N(C)C)C1CC1)C 35390,c1(C(C(N2C(C(N)=O)CC2)=O)NC(c2ccco2)=O)ccc(Cl)cc1Cl 35391,C1(C(N2CCC(CNC(CCS(C)=O)=O)C23CC3)=O)COc2cc(F)ccc2C1 35392,N1(C(c2cc(OCC)cc(F)c2)=O)CC2(CC(NC(=O)CCC3(C)CC3)CO2)C1 35393,c1(C(N2CCC(N(C(=O)CS(=O)(=O)NC)CC)CC2)=O)ccc2nccn2c1 35394,C1(OC)CC(NC(c2ccccc2C(N)=O)=O)CN(C(=O)CNC(N)=O)C1 35395,c1(C(=O)NCCC2(O)CN(C(C(COC)O)=O)C2)cccc2c1CNC2=O 35396,c1(NC2CCN(C(CC3C(=O)NC(=O)N3)=O)C2)ncnc2c1CCC2 35397,CC1C2C(CCN2C(=O)C=CCN2CCCC2)CN1C(=O)CCOC1CCOC1 35398,c1(C(N2CC(C=C)(CC(=O)NCCOC3CCOC3)C2)=O)ccc([N+](=O)[O-])[nH]1 35399,C1(C(=O)NC(C(C)NC(C2CC2c2cccc(F)c2)=O)(C)C)CCCC(=O)N1C 35400,C(=O)(C1=CC2CCCCC12)N1CC(CNC(=O)CC2(O)CCC2)C(C(F)(F)F)C1 35401,c1(NC(c2c(C)ccs2)=O)ccc(C(=O)OC2CC3CCC2CC3)c(F)c1 35402,N1(C(c2cc(C)ncc2C)=O)CC2CCCC(C1)N2C(c1cccc(N)c1O)=O 35403,C1(C(=O)NC2(NC(C3CCCN(C(N(C)C)=O)C3)=O)CC2)CCC12CCOCC2 35404,C(=O)(C(F)CC(CC)CC)NC(C(=O)NCCc1cc(CC)no1)(C)C 35405,C(=O)(C1CCCc2sc(=N)[nH]c21)N(CC(CNC(C(CCC)C)=O)(C)C)C 35406,N1(C(CC=C)=O)CC(C)(C)CC1CC(=O)NC(C)C(O)C(F)F 35407,N1(C(C(C)Sc2nncs2)=O)CCn2c(nc3c2CCCCC3)C1 35408,C1(C(N(C(CNC(c2cc(C(C)(C)C)no2)=O)C2CC2)C)=O)CCCSS1 35409,C1(N(C(c2ccc(C(C)C)cc2)=O)CC)CCCN(C(C2(C3CC3)CC2)=O)CC1 35410,c1(C(=O)NC2COCC2NC(C23CSC(C2)C3)=O)n[nH]c2cccnc12 35411,N1(C(Cc2ncc(CC)[nH]2)=O)CC(CCNC(=O)CC(=O)NC2CC2)OC(C)C1 35412,C(C(C(F)(F)F)N1CCN(C(=O)CC2C=CCC2)CC1)NC(CN(C)CCO)=O 35413,c1(C(N2CC(N(C(=O)CC3CC(C(F)F)C3)C)C2)=O)coc(Cl)c1 35414,C1(C(N2CCC(CN(C(=O)CN3CCC(C)(C)C3)C)CC2)=O)CCCCC12CC2 35415,c1(C(=O)NCCC(C)NC(c2ccc(Cl)o2)=O)oc2ccccc2c1CO 35416,c1(N2CCC(NC(c3cnn(CC)c3C)=O)C2)cccc(F)c1C#N 35417,C1(C(N2CC(C)(NC(c3cn4c(n3)CCC4)=O)C2)=O)CCC(S(C)(=O)=O)CC1 35418,C(=O)(C(F)CCC(C)(C)C)N(C1CCN(C(CCCC)=O)CC1)CC 35419,c1(CCC)ccc(C(=O)NC2COCCC2NC(C2CC(F)C2)=O)cc1[N+](=O)[O-] 35420,C(=O)(CC(O)C(C)(C)C)NC1CCC(NC(C2ON=C(C)C2)=O)CC1 35421,CCCCC(C(=O)NCC=CCSC)NC(=O)CCC(N)=O 35422,c1(CNC(c2nnnn2C2CC2)(CSC)C)nnc(C2CC2)n1C 35423,c1(C(N2CCCC(CC(=O)Nc3nccc(C)c3)C2)=O)cc(Br)cnc1O 35424,c1(C(=O)NC2CN(C(C3(O)CCOC3)=O)CC2O)cc(F)cc(Cl)c1 35425,N1(C(C(C)(C)SC)=O)CCN(CCCNC(=O)C(=Cc2cccs2)C)CC1 35426,c1(CC(=O)NC2CCCCN(C(=O)Cc3cn[nH]c3)CC2)cccc2nsnc12 35427,C(=O)(C1=C(Cl)CCOC1)NCC(C)(C)OCC(=O)Nc1c(CC)cccc1 35428,c1(C(N2CCN(C(=O)CC3CC(F)C3)C(C3CC3)C2)=O)ccc2c(c1)COCO2 35429,CCCC(C)(O)CC(=O)N1C2CCC(C2)C1C(=O)NCCCc1ccccc1 35430,N1(C(CCC(C)C)=O)CCOCC2(COCCN2C(=O)C2=CC3CCCC23)C1 35431,c1(CC)ccc(C(=O)NC2CCC(NC(C3(F)CC3)=O)C2)[nH]1 35432,C(C(CC(C)(C)C(=O)OC)NCc1cn(-c2cc(C)cc(C)c2)nn1)OC 35433,C12(CNC(C(C(C)C)C)=O)CCC(CN(C(=O)CCCc3n[nH]c(=N)s3)C1)C2 35434,Cc1[nH]c(C(=O)NCCCO)c(C)c1C(=O)Nc1cnc(Cl)cn1 35435,C(=O)(CC1=NNC(=O)C1)NCC1CCN(C(c2cnc(CC)[nH]2)=O)CC1C 35436,C1(C2CC2)(CNC(C=CC)=O)CCN(C(c2c(C)nnn2-c2ccccc2)=O)C1 35437,c1(OC)cnc(F)cc1C(=O)NCC(C)(CO)NC(=O)C=Cc1ccc(O)cc1 35438,Cc1cccc(C(N2CC(CC(C)NC(=O)COC3(C)CCC3)C2)=O)c1Cl 35439,C(=O)(C1=NOC2(CCN(C(C3C4C=CSC34)=O)C2)C1)Nc1cc(C(C)C)no1 35440,N1(C(C(C)n2cnnn2)=O)CCN(C(=O)C#CC2CC2)C(CC(F)F)C1 35441,c1(C(=O)NC(CC)CNC(=O)CCc2ccc(F)nc2)cncc2cccnc12 35442,C1(C(=O)NCC2(NC(c3cc[nH]c3)=O)CCC2)CC12CCSCC2 35443,C(=O)(C(O)C(C)OC)N(C1CCN(C(C2(CF)CCC2)=O)CC1)CCC 35444,c1(CC(N2CC(C(C)(C)O)(CNC(CSC)=O)C2)=O)ccc(S(=O)(=O)NC)cc1 35445,C#CC1(O)CN(C(=O)CN(C(=O)CC2CC3(CCC3)C2)C2CCC2)C1 35446,C1(CC)C(C(=O)NCC2(O)CCN(C(c3ccc(CO)cn3)=O)C2)CCN1C 35447,c1(OC)ccc(C(N2CCC(C3CCCN3C(c3ncoc3C(C)C)=O)C2)=O)o1 35448,c1(CC)nn[nH]c1CNC(c1csc(CNC(C2COC(C)C2)=O)c1)=O 35449,c1(C(=O)NCC(CC)NC(=O)CCC(C)OC)ccc(N)c(CC(C)C)c1 35450,C(=O)(CCCCN(C)C(C1CC(F)C1)=O)NC(c1nnc(C)o1)C 35451,C(=O)(C1=NNC(=O)C1)NCC(CC(=O)N(C(CC(CC)C)C)C)O 35452,c1(CNC(C(C(C)O)NC(=O)CC(C)(C)O)=O)ccc(C#N)cc1 35453,c1(C(=O)NCCC2(OC)CN(C(=O)CC3(C)CCC3)C2)cncc2sccc12 35454,c1(CCC(=O)NC2CC(NC(C=CS(C)=O)=O)C2)nnc(S)nc1O 35455,CC1(C)CC2(CC2C(=O)NCC2(NC(c3ccc(F)c(C(F)F)c3)=O)CC2)C1 35456,C(=O)(CCC(C)(C)F)NCC(CCNC(C1N(C(CC(C)C)=O)CCCC1)=O)O 35457,C1(NC(=O)CSc2ccsc2[N+](=O)[O-])CCN(C(=O)COC2CCC2)C12CCC2 35458,c1(CC(=O)NC(C2CCCN(C(=O)CC3(O)CC3)C2)C)ccc(F)c(F)c1 35459,C1(C(N2CCC(NC(C(CC)=CC)=O)C(C)C2)=O)CCCC2CCCN12 35460,CC1(C)CCCC(C(=O)NC2CCCC23CN(C(c2snc(Cl)c2Cl)=O)C3)CC1 35461,CC(C)(CCC(=O)NCc1nc(=O)o[nH]1)NC(=O)CCc1cccnc1 35462,c1(CC(C(=O)NCCC2(NC(CC3CC(OC)C3)=O)CC2)C)ccc(F)cc1 35463,N1(C(c2nc(C)nn2C)=O)CCC(C2(O)CN(C(=O)C(C)S(N)(=O)=O)C2)CC1 35464,N1(CC)C(=O)CCC1CC(=O)N(C)CCOCCNC(=O)CN1CSCCSC1 35465,C1(C)(CCC(=O)NCCCN(C(C)C)C(C2CC(F)(F)C2)=O)CCC(=O)N1 35466,n1(CC(=O)NC2(C)CC(NC(C3(CC)CCNC3=O)=O)C2)c([N+](=O)[O-])cnc1C 35467,O=CCCC(=O)N1CC(NC(c2ccnc(C(=O)O)n2)=O)C(F)C1.N1CCCC1 35468,C12(C(N3CCCC(NC(COCCCC)=O)C3)=O)CC3CC(CC(C3)O1)C2 35469,Cn1cc(C(CO)NC(=O)CNn2cc(-c3cnn(C)c3)nn2)nn1 35470,c1(C(=O)NC2C(C(C)C)N(C(=O)CCN3CCC(F)C3)CC2)cc2c(s1)CCC2 35471,CC(C)S(=O)(=O)CCCN1CC=CC(NC(c2coc(Cn3cccn3)c2)=O)C1 35472,C(=O)(CC(C)(C)N(C(=O)CC1CCC(=O)N1C)C)NC(c1ccccn1)CC 35473,C=CC1CN(C(=O)Cn2cc(C3CCC3)nn2)CC1NC(c1cc(C)c(C)[nH]1)=O 35474,N1(C(C(C2CCOCC2)OCC)=O)CCC2C1CCCN2C(c1cnc(O)s1)=O 35475,C=C(Cl)CC(C(=O)NOC(C)C(=O)OC)NC(=O)CC1CN(C(=O)NC)C1.CCC 35476,C1(CC=C)(C(=O)NCCC(O)C2CCCC2)CCN(C(=O)C=Cc2cocn2)C1 35477,Cc1ccc2n[nH]cc2c1C(N1CC(C)(NC(c2cnc(O)c(Br)c2)=O)C1)=O 35478,N1(C(CC(=C)C)=O)CC2CCC(N=c3ccc(C(=O)OC)c(OC)[nH]3)CC2C1 35479,N1(C(c2c(C)nc(CC)s2)=O)CC(CNC(c2ccsc2C#N)=O)CC1(C)C 35480,C(=O)(C1CCCc2c[nH]nc21)N1CC2C(NC(CN3C(=O)CC(C)(C)O3)=O)C2C1 35481,c1(CC(=O)NC(C)CCNC(=O)C(C)C2CCCO2)ccc2nonc2c1 35482,C1(NC(C=COCC)=O)CC2CC(C1)CN(C(=O)COc1cc(F)cc(F)c1)C2 35483,C1(C(=O)NC(C)CCOC)(CC)CCCN(C(c2cc(CO)nn2C)=O)C1 35484,c1(CC)cc(C(N2CC(NC(=O)C(C#N)C3CC3)C(O)C2)=O)ccc1F 35485,c1(C(=O)OC)ccc(C(=O)NC2CCC(NC(=O)CS(N)(=O)=O)CC2)nc1 35486,c1(CCC(=O)NC(CC)CNC(C2CCC(F)(F)CO2)=O)nc2ccccc2o1 35487,C(C1(C)COC1)=CC(=O)N(CCN(C(C1(Cl)CC1C(=O)OC)=O)CC)CC 35488,N1(C(C2CCCN(CC)C2)=O)C2CCC(C2)C1CNC(c1ccc(O)nc1)=O 35489,N1(C(C)=O)CC2(COC(CNC(c3cnn(CC(F)(F)F)n3)=O)C2)C1 35490,N1(C(C(C)(C)C2(O)CCC2)=O)CCCC(Cn2ccnc2)C1 35491,CCC(CC(C)C)C(=O)NCC1(O)CN(C(=O)Cc2ccn(CC(F)(F)F)n2)C1 35492,O=C1CCc2cccc(C(=O)NC3CCCC3CNC(c3coc(CO)c3)=O)c21 35493,C1(C)(NC(C(CCCNC(C=C(C)C(F)F)=O)O)=O)CCC(=O)NC1=O 35494,C1(CC#C)CCN(C(=O)CCC2CCN(C(c3ncn(C)n3)=O)C2)C1 35495,c1(C(=O)NC2C(C(=O)NCc3c(C)nccn3)CCC=C2)ccn(C)c(=O)c1 35496,C1(C(NOC(C(=O)OC)(C)C)=O)CC2CC1CC2NC(=O)C(=O)NC(C)C 35497,N1(C(C(Cn2ccnn2)NC(=O)CNC(C2CCCO2)=O)=O)CCC(O)CC1 35498,C=C1CCN(C(=O)Cc2ccnn2C)C(C(=O)NC2(CC)CCCCC2)C1 35499,C1(CC)CN(C(=O)C=Cc2cccnc2)CCN1C(=O)CSCCOC 35500,N1(C(c2c(C)ncs2)=O)CCCC2C1CCCN2C(C1CCC(N(C)C)CC1)=O 35501,c1(NC(C(C2CN(C(C(COC)O)=O)C2)OC)=O)cncc(N2CCCC2)n1 35502,N1(C(C2CCN(C(c3n(CC)ccn3)=O)C23CC3)=O)CCC(O)CC(C)C1 35503,N1(C(C(CCOC)OC)=O)CCN(C(=O)CCCSC)C(C)C1 35504,CC1CS(=O)CCN1C(C1CCCC(NC(=O)CCc2nccs2)C1)=O 35505,C12(C(=O)NCC(C(C)C)CO)COCC1CN(C(c1cc3ncccn3n1)=O)C2 35506,C(C(=O)N1CC(CCNC(=O)CCSC)C1)(C(C)C)NC(=O)OC 35507,c1(C(=O)NCCCC(C)NC(CCNC(COC)=O)=O)ccc(C)nn1 35508,Cc1ncc(C#N)cc1NC(c1conc1CNC(C1(C)CCC(C)C1)=O)=O 35509,N1(C(CCC(=C)Cl)=O)CCC2CN(C(C3(C)CCCNC3=O)=O)CC2CC1 35510,C1(CC)CN(C(=O)CC2CS(=O)(=O)C2)CCN1C(=O)COc1cnn(C)c1 35511,C(=O)(CC(C)CNC(=O)C(C)c1ccco1)NCc1n(CC)cnn1 35512,C(CC(C)C(=O)N1CCN(CCNC(=O)Cc2n[nH]c(=NC)s2)CC1)=CC 35513,CC(C)CCC(F)C(=O)NC1(CCC(=O)N(C)Cc2ccsc2)CCCC1 35514,c1(OC)ncnc(C(=O)NC2(C)CN(C(C3CCOC(=O)CC3)=O)C2)c1F 35515,N1(C(C2CCC(C)=CC2C)C(=O)NCC(=C)C)CCCC2OCCC2C1 35516,CCC(Cc1ccccc1)C(=O)NCC1(F)CN(C(=O)C(c2cnccn2)C)C1 35517,CCCC(CC)C(=O)NCC(C(C)(C)C)NC(c1cc(=O)c(Br)c[nH]1)=O 35518,N1(C(CC2CC(=O)OC2)=O)CC=CC(C(=O)NC2CC(CO)C3CC23)C1 35519,CC(CC(C)NC(=O)CS(=O)(=O)NC1CC1)N=c1[nH]c(Cl)nc2ccccc12 35520,CC1(C(=O)NCC2CC(NC(C3CC(=O)N(O)C3)=O)C2)CS(=O)(=O)C1 35521,C1(CCCNC(c2ncn(C)c2)=O)CCN(C(C2(CO)CCCCO2)=O)CC1 35522,C(CC(=O)NC(C(N)=O)C1CC1)(C1CC1)NC(CSC)=O 35523,CCCC(C)(CCCNC(N1CCCC(OC)C1C)=O)C1OCCO1 35524,N1(C(c2c(C)[nH]cc2)=O)CCCCC(C(=O)NCCc2ccnc(O)c2)C1 35525,c1(C(=O)NC2CC(C)(NC(CC(=C)Br)=O)C2)c(O)nnc2c1CCC2 35526,C(C)(CCCNC(=O)C=CCOC1CCOCC1)NC(CSCCCC)=O 35527,C(=O)(NNc1cccc2c1CCCC2)C1(C(=O)OC(C)(C)C)CC(F)C1 35528,N1(C(c2cc(Br)cs2)C(=O)NCCC2CC2)CC2CCCCN2c2ccccc21 35529,c1(C(=O)NCCCCCN(C(CN2C(C)CCC2C)=O)C)cc2occc2n1C 35530,c1(C(N2CCCC(CNC(c3on(C)c(=O)c3)=O)CC2)=O)c(F)ccc(F)c1N 35531,N#CC1(C(N2CCN(C(C3(S(N)(=O)=O)CCC3)=O)CC2)=O)CC2CC2C1 35532,N1(C(C2CCN(CC(C)C)C2)=O)CCN(C(=O)C2=CSCS2)CC1C1CCC1 35533,Cc1cc2[nH]c(C(=O)NC3CC(C)CN(C(C4CC5COCC5C4)=O)C3)cc2s1 35534,CC(=O)CC(C)(C)C(=O)N1CCC(C)C(CNC(C2CN(C)CC(C)O2)=O)C1 35535,C1(C(=O)Nc2cn(C)nc2Cl)CC2CCC1N2C(C1CC(C)(F)C1)=O 35536,CN=c1[nH]c(=NCCCc2nc(C)cs2)[nH]c(=NC2CCOC(C(C)C)C2)[nH]1 35537,c1(C(N(CCCCN(C(CCn2c(C)ncc2)=O)C)C)=O)ccc(F)c(Cl)c1F 35538,c1(CC(N2C3CCC2CC3)=O)cc2ccccc2s1.c1(OC)cc2c(cn1)NC2=O 35539,N1(C(c2c(C)ccnc2)=O)CCCC(C)C1CNC(=O)C(F)C1CCOC1 35540,c1(C(N2CCN(C(c3ccc(C(C)=O)nn3)=O)C3C2C3)=O)c[nH]c2ccccc12 35541,N1(C(C2(C(=O)OCC)CCCC2)=O)CC2(CCC2NC(c2cn(C)nc2O)=O)C1 35542,C1(CNC(C2C(C)(C)CC2)=O)CCCN(C(C2(c3ccc(Cl)cc3)CC2)=O)C1 35543,N1(C(CN(C(=O)C(C)c2cccs2)CC#C)=O)CCC(C)(CO)C1 35544,C(=O)(C(C)C(O)CC(C)C)N1C(C)(CC(=O)Nc2c(F)ccc(C)c2)CC1 35545,c1(OC)ccc(CC(=O)NCCC(O)CNC(C2CNC(=O)N2)=O)cc1O 35546,C=CCC(CNC(C1(C)CC(=C)C1)=O)NC(c1csc(C2CCCCC2)n1)=O 35547,C=C(Cl)CC(C(=O)NC(c1ncc(C)o1)C)NC(=O)Cc1ccn(CC)n1 35548,C1(NC(c2cc(O)nc(O)n2)=O)C2CC3CN(C(C4CC45CC5(F)F)=O)C1C3C2 35549,Cc1ccc(C(=O)NCC(C)(CO)NC(=O)CC2CCC2(C)C)c(O)n1 35550,c1(OC)c(C(N2CCCCC(Cn3cc(C4CCC4)nn3)C2)=O)ccc(Cl)c1Cl 35551,c1(OCC)cc(C(N2CCC(=CC(=O)Nc3ccccc3C)CC2)=O)cc(F)c1 35552,Cc1ccc(Cl)c(C(=O)NCCNC(c2ccc(CN=[N+]=[N-])cc2)=O)c1N 35553,N1(C(CCCOC)=O)CCC(NC(=O)CSc2nc3ccccc3s2)C(C)(C)C1 35554,C1(NC(C(C)NC(C2CNC(=O)N2)=O)=O)(CO)CC2CCCC12 35555,CCCCCCCCCC(=O)NCC1CC2(CC2)CN1C(=O)C(O)C(F)F 35556,N1(CCNC(c2nc(C(C)C)oc2)=O)CCCN(C(C2CC2(F)Cl)=O)CC1 35557,CC1CC(C(F)(F)F)n2nc(C(=O)OCC3CC4(CC4)C(=O)O3)cc2N1 35558,n1(CC=C)nnnc1C(c1cc(C(F)(F)F)cs1)NCC(C)OC 35559,Cc1nc([N+](=O)[O-])cn1CC(=O)NCCC(C(C)C)NC(C1CCOC(=O)N1)=O 35560,C1(NC(C(n2c(C)nnn2)Cc2ccc(F)cc2)=O)COC2(CCC2)CO1 35561,c1(C(=O)NCC2(CNC(C(C(C)C)OC)=O)CC23CCC3)ccc(Cl)c(F)c1O 35562,O(C1CCCc2cc(Br)ccc21)C(=O)NC1Cc2c(cn(C)n2)CC1 35563,C(=O)(C(O)CCCc1ccccc1)N(CCNC(C1CCN(C)C1=O)=O)C1CC1 35564,N1(N2CCn3c(O)nnc3C2)CC2C(SCCNC=O)C3CCC2(C1)O3 35565,c1(NC(C2C(CNC(C=C(COC)C)=O)CCCC2)=O)ccc(C)nc1C 35566,C1(NC(c2c(C3N(C(CS(CC)=O)=O)CCCC3)n[nH]c2)=O)(CO)CC2CCCC12 35567,c1(C(=O)NCC(C)CNC(C23CC(C)(C2)C3)=O)cc2c(o1)CCCNC2=O 35568,C1(CNC(c2c(N)c(Cl)ncc2)=O)CCC2(CCC2)C1NC(=O)C=C1CC1 35569,N1(c2n(CCOC)c(CO)nn2)CC(CC(=O)NC2(CF)CCC2)c2ccccc21 35570,Cc1cn2cccc(C(N3CC(C4(NC(=O)Cc5csc(S)n5)CC4)C3)=O)c2n1 35571,C1(C(=O)NCC2C3CN(C(=O)C(C4CCCCCC4)O)CC23)(CC)CCCCC1 35572,n1(CC)cccc1C(=O)NC1CC1NC(=O)C(c1ccccc1)OCCC(C)C 35573,C1(C(=O)NCC(CC(F)(F)F)NC(c2c[nH]c(=N)s2)=O)CC2CCCC(C1)C2 35574,N1(C(C(CC=C)NC(C)=O)=O)CCC(C)N(C(=O)CSC(C)(C)C)CC1 35575,CN1CCN(C(=O)CCc2cc(F)ccc2Br)C(CNC(=O)C(N)=O)C1 35576,c1(OC)ccc([N+](=O)[O-])cc1-n1cc(CN(C(=O)C(C2CCC2)OC)C)nn1 35577,CCCS(=O)(=O)CC(=O)N1CCC(O)(c2cncnc2)CC1 35578,N1(C(c2c(OC)ccnc2)=O)CCCC(NC(=O)CC(C)(C)C#N)C1C 35579,N(C(=NCCCSC)NCC1CC2CCC2C1)C(C#C)COC 35580,CCCCCCCCNC(=O)C(=O)NC1CN(C(=O)C(C)SC)CCC1F 35581,n1(CC(N2CCN(C3CCCN(C)C3)CC2)=O)ncc(Cl)c(Cl)c1=O 35582,Cc1ccc(Cl)cc1C(=O)NCC(O)CN(C(=O)CN1CCC(C)C1)C 35583,CC1CN(C(C2CC(O)(CNC(C3(C)CCC3)=O)C2)=O)CC(C)(C)C1 35584,CC1(NC(C23CC(CN2C(C2(CCN=[N+]=[N-])CC2)=O)C3)=O)CCOC1=O 35585,C1(CNC(C(c2ccc(C)o2)C)=O)CN(C(=O)C=Cc2cccs2)C(C)(C)C1 35586,C1(N(C)C(c2ccc(Br)o2)=O)CN(C(c2ccncc2)=O)CC1O 35587,c1(C(N2CCC(C(N(CCC(=O)OC)C)=O)C2)=O)ncc(F)cc1F 35588,C(N=c1nc(N2CCCC(Cn3ccnn3)C2)cc(C)[nH]1)C1(OC)CCC1 35589,N1(C(C2C(C(=O)OC)C2)=O)CCN(C(c2csc(C(C)(F)F)n2)=O)CC2(CC2)C1 35590,c1(C(=O)NCCC(C)N(C(Cc2c(C)n[nH]c2)=O)C)cc2c(cnn2C)nc1C 35591,C1(CC)CN(C(=O)C(=O)NC23CC(C(F)F)(C2)C3)CCN1C(C)=O 35592,N1(C(C2CC(C)SCC2)=O)CC(NC(C2COC(C)(C)C2)=O)CC(C)(C)C1 35593,C=Cc1cnc(NC(N2CC=CC(O)C2)=O)cc1F 35594,N1(C(c2c(CC)noc2)=O)CC(CNC(c2cccc(C)c2)=O)CCC1C 35595,c1(C(N(C(CC(=O)OCC)c2ccccc2)CCC)=O)ccc(CCOC)o1 35596,c1(C(=O)NCc2occ(C(=O)NCC(C(CC)C)C)c2)ccnc(C)c1N 35597,c1(C(N2C(C(C)NC(CCCCCC=C)=O)CCC2)=O)cc(N)c(F)c(F)c1Cl 35598,c1(C(N(CC(C)NC(=O)CCOCC(F)(F)F)CC)=O)cncc(Br)c1 35599,C(c1cn(CCCN(C)C(C2CCN(c3ccc(Cl)cn3)CC2)=O)nn1)=CC 35600,C1(C(N(C(CNC(C(C)O)=O)Cc2ccccc2)C)=O)CCC(F)CC1 35601,C12(C(N3CCC(NC(c4cc(C)cc(O)c4)=O)CC3C)=O)CCC(C)(CC1)OC2 35602,N1(C(C23N(C(C(=CC4CCCC4)C)=O)CC(C)(C2)C3)=O)CCC2CC1C(=O)O2 35603,C1(NC(CC(C)F)=O)CC(F)CN(C(c2cncc(N3CCCC3)n2)=O)C1 35604,Cc1ccc2sc(C(N3CCN(C(=O)C(C)C4CCOC4)CCC3C)=O)cc2c1 35605,N1(C(c2c(C)nc(C)o2)=O)CC2CCCC(C1)N2C(=O)C(C)n1ccnc1 35606,c1(CC(=O)NCCOC2CN(C(CC(C)OC)=O)C2)cnccc1Cl 35607,C(=O)(CCC(=O)N1CC(CCNC(C2(SC)CCC2)=O)C1)Nc1nnc(CC)s1 35608,C12(C(N(CCN(C(C3CC3(C)C(C)C)=O)CC)CC)=O)CC(C)(C1)OC2(C)C 35609,CC1(C)CC(CC(=O)Nc2ccnc(C3CC3)c2)C(=O)O1 35610,C1(NC(=O)CCC(F)(F)F)CCCC2CN(C(=O)CC3CCOC3)CC12 35611,C1(Nc2ccc(CC)cc2)CC2c3ccccc3C1c1ccccc12 35612,Cn1nnc(CNC(=O)C(c2ccccc2)NC(n2cnnn2)=O)n1.c1cc(F)c[nH]1 35613,N1(C(c2c(C)occ2)=O)CCC2CC(CNC(C3CCC(C)CC3)=O)CCC2C1 35614,CC(C)CC(C(=O)NCCc1noc(=O)n1C)ONC(=O)C1(N(C)C)CC1 35615,C1(CC(C)C)(C(N(C2CC(NC(CCC=CC)=O)C2)C)=O)CCNC1=O 35616,C1(NC(c2cccc(F)c2OCCF)=O)CN(C(=O)COC(F)F)CCC1CO 35617,c1(C(CC)O)nc(C2CCC(=O)N2C)n(-c2nc(C)nn2C)n1 35618,N1(C(CCCCOCCC=C)=O)CCN(C(c2ccnc(C)c2)=O)C(C)C1C 35619,C1(F)(C(=O)OCC)CN(C(=O)C(=O)c2ccco2)CC1(C)C(F)(F)F 35620,N1(C(c2onc(CC)n2)=O)CC2(CCN(C(=O)Cc3cccs3)CC2)C1 35621,c1(NC(CN2C(CNC(C(C)NC(c3ccoc3)=O)=O)CC2)=O)cc(Cl)c(Cl)n1C 35622,c1(OC)ccc(F)cc1CC(=O)NC1CCN(C(=O)Cc2ccc(C)o2)C12CC2 35623,N1(C(C(=O)NC(CC)C)=O)CCOCC(CNC(c2ccc(C)[nH]2)=O)C1 35624,C1(C(=O)NCC(CC=C)NC(c2cc(CCC)oc2C)=O)CC2C=CC1C2 35625,CC(C(=O)NC(C(=O)NCC1(CO)CCC1)c1cccs1)OC1CCCC1 35626,C(=O)(CCCC(C)(C)C)N1CCC(CN(C(=O)Cc2cn3ccsc3n2)C)C1 35627,Cc1cc(O)nnc1C(=O)NC(C)CCNC(=O)C(C)(C)c1cscc1Cl 35628,c1(CC)c(NC2CCN(C(C3(F)CCOC3)=O)CC2C)nc(C)nc1Cl 35629,N1(C(c2nnn(CC)c2C)=O)CCC(C2(NC(c3[nH]ccc3C)=O)CC2)CC1 35630,[N-]=[N+]=NCCCC(=O)NCC1(O)CC(CNC(=O)CCc2csc(=N)[nH]2)C1 35631,c1(C(N(CCOCCN(C(c2cc(C)c(C)[nH]2)=O)C)C)=O)cc2ncccc2o1 35632,C1(CCC#C)CCCN1C(=O)C(=O)NCC1CCCN1c1cccnn1 35633,N1(C(C(CC)OCC)=O)CCC2(CCCN2C(c2cc(C(F)F)no2)=O)CC1 35634,n1(CC)nc(C)cc1C(=O)NCC1CC1NC(=O)C(C)(C)n1ccc(C2CC2)n1 35635,C1(CC)CCN(C(c2ccc(SC)s2)=O)C1C(=O)Nc1cnn(C)c1SC 35636,N1(C(c2ncncc2Cl)=O)CCC(CNC2C(C)(C(F)F)C2)C(O)C1 35637,N1(C(c2c(C)nc(C)o2)=O)CC2(COC(CNC(c3csc(S)n3)=O)C2)C1 35638,N1(C(c2cnn(C(C)C)n2)=O)CCC2CN(C(c3cnccn3)=O)CCC2C1 35639,C(=O)(CCS(=O)(=O)C(F)(F)F)NCCCC(C)NC(C(CC)(C)OC)=O 35640,C=CCC(C)C(=O)NCC1(C(=O)NCCOC(C)=O)CC=CC1 35641,CC(C)(C(=O)NCC(O)CNC(C1CC(n2ccnn2)C1)=O)C(F)(F)F 35642,Cc1c(F)ccc(C(=O)N(C2CCC(NC(C3CCCCC3C)=O)CC2)C)c1C 35643,C1(NC(C(C)OCCCCCC)=O)C=CCN(C(=O)CC2(C3CC3)CC2)C1 35644,Cc1cc(C)c(C=CC(=O)NC2(CO)CCN(C(=O)C(O)C3CC3)CC2)cc1C 35645,C(=O)(C1=CCC2CCC1N2C(C1(C)CCC1)=O)N1CCC(C)(O)CC1 35646,N1(CC(=O)NC2(CN(C)C(c3cnn(C)c3)=O)CC2)CC2CC2C1 35647,c1(C(=O)NC2CN(C(C(CCCC)N(C)C)=O)CC2C)c(Cl)ccc2ccoc12 35648,c1(NC(c2cc(CC)on2)=O)ccc(S(=O)(=O)N(CCOC)CC)cc1 35649,CCC(CC)CCCC(=O)N1CC2CCC1CC2NC(C1C=CC=CC=C1)=O 35650,N1(C(c2scc(CNC(C(C=CC)O)=O)c2)=O)CCc2c(cnn2C)C1 35651,CC(=O)CCN=C(NCC1CCCCS1)NCC(C1COC(C)(C)O1)(C)O 35652,C12(CNC(C3CCN(C(C4CCNC4=O)=O)CC3)=O)CCC(CC1)O2 35653,C(N=c1nc(C(=O)OC)c(Cl)c[nH]1)C1CCC(NC(C(CCC)(C)O)=O)C1 35654,c1(OC)cc(C(=O)NC(CNC(C2CCCC23CC3)=O)C2CC2)c(F)cc1N 35655,C(=O)(C(C)C(O)CC)N(CCOCCCN(C(CCOCC=C)=O)C)C 35656,C1(c2n(C)ccn2)CCN(C(=O)NCC2CC(OC3CC3)C2)C12CC2 35657,c1(C(=O)NC2CN(C(C(CC)OC3CCCCC3)=O)CC2F)cc2sccc2[nH]1 35658,c1(C(=O)NCC(CC=C)NC(=O)CN2CC3CCC2C3)c([N+](=O)[O-])cnn1CC 35659,C1(CNC(c2c(C(C)C)noc2)=O)CN(C(C2CC3CC3C2)=O)CCC1C 35660,Cc1cc(C(N2CCOC(C(C)NC(C3CCCCO3)=O)C2)=O)cc(C)c1F 35661,C1(NC(C(CC#C)C)=O)CS(=O)(=O)C2CN(C(=O)CNC(=O)NC3CC3)CC12 35662,C1(C(=O)NC2CC(NC(C3CC4(CC4)C3)=O)C2)CCC12CCCO2 35663,c1(C(=O)NC2C(NC(c3nncc(OC)c3)=O)COCC2)cc(C)c(Cl)cn1 35664,S(=O)(=O)(c1cccc(C(F)(F)F)c1)NC(C1CCC(Nc2c(C)cncn2)C1)=O 35665,C1(N(C)C(C2(CC3(C(N)=O)CCCC3)CC2)=O)CCC(n2cc(C3CC3)nn2)C1 35666,N1(C(=O)CO)CCC2(CC1)CN(C(c1ccc3nn[nH]c3n1)=O)CCO2 35667,c1(C(=O)NCC2CC(NC(c3c(CC)ncs3)=O)C2)ccc2c(c1)C(=O)CCO2 35668,C1(c2nnnn2C2CC2)(NCCNC(=O)OC)CC(C)(C)C1.n12cc(cn1)C2 35669,CC1CC(CNC(=NCCN2CCNC(=O)C2)NCC(F)F)CC(C)O1 35670,N#Cc1ccncc1NCc1ccc(C(=O)NCc2ccc(Br)cc2Cl)cc1 35671,C1(C2CCOCC2)(C(N(C2CCC3CC23)C)=O)CC1 35672,C(C(C(=O)NCCN(C(=O)C(C)(C)n1ccnn1)C)C(C)(C)C)OCC=C 35673,C1(=O)CCCC(=O)NCCCCN1CC.c1(C(=O)NCC)ccc(CO)cn1 35674,Cc1c(C(F)(F)F)n[nH]c1C(=O)NC(C)CN(C(=O)C(n1cc(Cl)cn1)C)C 35675,C(=O)(CCCCCC#N)N1C(CNC(c2cc(C)n(C3CC3)c2C)=O)CC(F)C1 35676,c1(C(=O)NCC#CC(=O)N(C)Cc2ccncn2)cccn(C)c1=O 35677,c1(CC)oc2ccccc2c1C(=O)NC1CS(=O)(=O)CC1NC(C1CCC1)=O 35678,c1(CNCC2N(CC(C)C)CCC2)n[nH]c2cc(F)ccc12 35679,c1(N2CCC(CN(C)C)C2)nc2c(c(=NCc3nc4ccccc4s3)[nH]1)COC2 35680,CCC(CCC(=O)NCCN(C)C)NC(=O)CN(CC(C)(C)C)C 35681,C1(CC(C)NC(C=C(COC)C)=O)CCN(C(=O)C(N2CCCCCC2)C)CC1 35682,c1(C(N2CCCCC2CC(N)=O)C(=O)NCC(C)C)ccc(C#N)cc1Br 35683,C1(CNC(CCC(C)OC)=O)CN(C(c2nnc(O)cc2O)=O)CC1(C)C 35684,c1(C(=O)Nc2cc(OC)no2)[nH]c(C)c(C(=O)Nc2ccccn2)c1C 35685,c1(C(=O)NCCCC(C)NC(c2cc(CC3CC3)on2)=O)cc[nH]c(=N)c1 35686,N1(C(C(CN=[N+]=[N-])NC(=O)C(C2CC2)C2CC2)=O)CC2CCC(O)C2C1 35687,n1(CC2(N(C)Cc3cc(OC)c(OC)cc3)CCNC2)cnc2ccccc12 35688,c1(CC)ncc(C(=O)N(C2CCCCC2)Cc2cccnc2)c(C)n1 35689,c1(OC)nccc(C(=O)NCc2occc2C(=O)NC(c2ccccc2)C)n1 35690,C1(F)(CNC(CN(C2CC2)CC)=O)CCCN(C(=O)CS(C)(=O)=O)CC1 35691,c1(C(=O)Nc2cncc(C(=O)NCC(N)=O)c2)cccc2ccnn12 35692,c1(OC)ccc(NC(C2CN(C(=O)C(=O)N(C)C3CC3)C2)=O)c(C)c1 35693,C1(C(=O)NCC(CNC(C(CC)=CC)=O)F)CCCC(NC(=O)OC(C)(C)C)C1 35694,N1(C(c2cc(N(C)C)ncc2)C(=O)NCC2CCOC2)CCCC(C)(C)CC1 35695,c1(CC(N2C(C)CC(NC(CC(CC)C3CC3)=O)C2)=O)ccc(O)c(C)c1 35696,C(=O)(CCCCCNC1CC1NC(c1ccc(Br)c(COC)c1)=O)OCC 35697,c1(CC(=O)N(CCOC)CCNC(C2CCC2)=O)cccc2cccnc12 35698,NC(=O)C1CN(C(C2CC3(C2)CC3(F)F)=O)c2ccccc21 35699,C(C)(CCC(=O)N1CCN(C2CCN(C(=O)C=C3CCC3)CC2)CC1)OC 35700,c1(C(=O)OCC)cc(Br)c(Cl)nc1N.c12cc(ccc1C)C(=O)N2 35701,C1(C(=O)NC(C)C)CCCCCC1NC(C1CC1(F)F)=O 35702,C(C)(C)(CC(=O)NC(C1CN(C(=O)CC2CCCS2(=O)=O)CCO1)C)SC 35703,c1(C(=O)NC(C)(C)CCNC(C2CCCCC2C(N)=O)=O)cc(N)ccc1Cl 35704,N1(C(CSc2cn(C)nc2)=O)CCC(CO)C(NC(=O)CCOC2CC2)C1 35705,c1(C(=O)N(C2CCCOC2)CCF)cc[n+]([O-])cc1 35706,N1(CC(=O)NCC(C(C)C)NC(=O)CC2CCCCN2C)CCC(=O)NC1=O 35707,c1(OC)cc(C(N2CC(C)(NC(=O)C(=Cc3ccccc3)C)C2)=O)cc(N)c1N 35708,C(=O)(CC(C(C)C)NC(C1CN(CC)CCO1)=O)N(CC=C)C 35709,C1(C(=O)NC2C(NC(C=CC(=O)OCC)=O)CC2)CC(=O)N(c2cnn(C)c2)C1 35710,C1(C)(OC)CCCN(C(C2CN(C(c3cnc(C)nc3)=O)CCO2)=O)C1 35711,C(=O)(CS(=O)(=O)CCC)N1CC(CCNC(CCC=CC)=O)OC(C)C1 35712,C1(N(C(=O)CN2CCSCC2)C)CCCC(NC(=O)C=CC2CCCC2)C1 35713,N1(C=O)CCCN(C(N)=O)CC1.Cc1ccc(CC(=O)NC2(C3CC3)CCC2)o1 35714,C12(CNC(c3cc(C)nn3C)=O)CCC1CCN2C(c1cnc(NC2CC2)s1)=O 35715,N(C(=NCCCF)NC1CCC(c2ccccc2Cl)C1)C1CCN(C(C)=O)CC1 35716,Cc1nc(NC(C2CC(C)CN2Cc2cnn(C)c2C)=O)cc(Cl)n1 35717,C1(CNC(C(CC=C)(C)C)=O)CC2CCC(C1)N2C(=O)CC1CC(C)C1 35718,Cc1nnc(NC2CCCCC2NC(=O)C(C)CC(N)=O)c(C#N)c1C 35719,c1(CN(C)C)ccc(C(=O)NC2COCC2CNC(=O)CN2CCCC2=O)o1 35720,C1(CC(=O)NC2CC(CCC(=O)N(c3cnc[nH]3)C)C2)CC2(CC2)CO1 35721,CC1=CC(C(=O)NC(C)C(=O)N(CCc2ccsc2)C(C)C)SC1 35722,CC1CC2CN(C(=O)CCCCNC(=O)CCNC(=O)CCC(CF)CF)CCN2C1 35723,N1(C(C2CCCN(C(C(C)CC3CC3)=O)C2)=O)CC2(COCC(=O)N2)C1 35724,N(C1c2ccccc2CC1(F)F)C(=O)NC1CC(C)NC(C)C1 35725,C(=O)(CCC1CCc2ccccc21)NCc1c(N(C)C)cc(C(=O)O)nn1 35726,C1(NC(=O)C=CC2CCCC2)CCN(C(C2CCCS2)=O)CC1F 35727,c1(NC(C(C2CC2)OC)C)[nH]c(=NCCc2ccsc2)nc2scnc12 35728,n12cnc(c1)C(=O)N(CCO)CC2.N#CCCSCC(=O)NCC1CC1 35729,N1(C(c2cc(CC)on2)=O)CCCN(C(=O)C(N2CCN(C)CC2)C)C(C)C1 35730,C(=O)(CC1=CCOCC1)N1CCC(N(C(=O)Cc2cccc(C#N)c2)CC)CC1 35731,C(N=c1cc(NCCSc2cc(F)ccc2Br)nc[nH]1)C1S(=O)(=O)CC1 35732,Cc1ccc2cc(C(N3CCCC(NC(c4sc(C)cc4Cl)=O)C3)=O)ccc2n1 35733,CCC(C)CCC(=O)NC1CC2(NC(c3cccc(N(C)C)c3)=O)COC1C2 35734,C1(N(c2n(C)nnn2)CCO)CCN(C(=O)NC2(CF)CC2)CC1.c1ccccc1 35735,c1(C(=O)NCC(CC)(C)NC(=O)Cn2cccc2)cccc(C2CC2)n1 35736,c1(CC(N2CC(OCCNC(C(C)=CC)=O)C2)=O)ccc2ncccc2c1 35737,N1(CC(=O)NC)CC2CCN(C(=O)CCCc3n[nH]c4ccccc34)CCC2C1 35738,c1(C(C(=O)NCCC)N(c2ccccc2)CC2CCOCC2)ccc(CC)cc1 35739,C1(C(N2CCC(C)(NC(c3ncc[nH]c3=O)=O)C2)=O)(CC)CCNC1=O 35740,N1(C(COCCC=C)=O)CC2ON=C(CNC(c3cccc4ncnn34)=O)C2C1 35741,CCCC(C)CC(=O)NCCC(C)NC(=O)CSc1cc(F)ccc1F 35742,c1(C(=O)NC(C2N(C(CCCC(=C)C)=O)CCC2)C)ccc2cc[nH]c2n1 35743,c1(OC)ncc(CN(C)C(=NCC2CCCNC2=O)NC2CCCC2)cc1Cl 35744,c1(N2C3CN(S(CCOC)(=O)=O)C(C3)C2)ncnc2cc(-c3ccccc3)sc12 35745,n1(CC(=O)NC(CC)CNC(=O)COCCSC)cnc(=N)[nH]1 35746,CN=c1[nH]c(=NCc2ccccc2OC(C)C)[nH]c(=NCCC2(C)CC2(Cl)Cl)[nH]1 35747,N1(C(C(COC)Cl)=O)CCC2(CCC2N2CC3CCC2C3)CC1 35748,C#CCCCCCC(=O)NC1(CCOC)CCN(C(=O)Cc2ccnc(C)c2)C1 35749,C1(NC(COCCC)=O)(CF)CCN(C(c2sc(C(C)C)nc2C)=O)C1 35750,N#Cc1cccc(C(=O)NC2CCN(c3ncnc4n[nH]cc34)CC2)c1Cl 35751,c1(C(=O)NCCC(C)NC(c2c(CC)nns2)=O)ccc(C#N)n1C 35752,N1(C(C(=O)NCC)CCC2CCC(F)(F)CC2)CCCC2CN(C)CCC12 35753,C1(NC(c2cnc(O)c(Br)c2)=O)CC12CCN(C(=O)CCCCC1CC1)CC2 35754,C(C(C(=O)N(C)CC1CCCCN1C(C1CCOC(C)(C)C1)=O)C(F)(F)F)OC 35755,Cc1ccc(C=CC(=O)NCCCNC(c2c(-c3cccs3)noc2C)=O)cn1 35756,c1(OC)ncc(Cl)cc1C(N1CCN(C(c2cc(C)co2)=O)CC1C(F)F)=O 35757,C(=O)(C(C)(C)CN(C(=O)Cc1ccsn1)C)NCCS(CC)=O 35758,N1(C(C2N(CC)CCC2)=O)Cc2ccccc2C(NC(=O)Cc2nnc(C)s2)C1 35759,CC1(C(N2CCC(O)(CCNC(C3CCC4(CC4)C3)=O)C2)=O)COC(=O)N1 35760,c1(OCC(=O)NC(c2nocc2C(N2CCC(CC3CC3)C2)=O)C)cccnc1 35761,c1(C(=O)NC(C)CCCCNc2ncc(C#N)cc2F)cnc2c(c1)ncn2C 35762,c1(NC(=O)NC(CC2CCCC2)CO)cccc2nc(O)nc(O)c12 35763,CC(C)CC(CNC(=O)CC1CCCCOC1)C(=O)NCC1(C)COCCO1 35764,N1(C(c2nn(NC(=O)CN(S(=O)(=O)CC)C)c(O)c2)=O)CCOCCC1.CCOC 35765,N1(C(C2(C)CCC2)=O)CC2COCCC2(NC(=O)CC2CCNC2=O)C1 35766,C1(C(=O)NCC(C2CC2)SC)CCN(C(=O)CC2CCCC(C)O2)O1 35767,C1(NC(CSCC#C)=O)CN(c2nnc(C(N)=O)s2)CC2(CC2)C1 35768,c1(C(=O)NCC2C(NC(=O)C=CC3CCC3)CC2)cnc2[nH]ncc2c1 35769,Cc1c(C(N2CC(NC(c3conc3C(F)(F)F)=O)C3(CC3)C2)=O)[nH]ccc1=O 35770,CC(C)C(O)C(=O)NCC(N1CCOC(c2ccco2)C1)=O 35771,N1(C(C(CCC)O)=O)CCC2(CC1)CC2C(=O)NC(c1ccc(Cl)cc1)C(=O)OC 35772,CN1CCC(C)(C(=O)NCC2CCN(C(=O)Cc3cn[nH]c3)CC2O)CC1 35773,c1(C(=O)NCCN(CCOC)C(C2CC(=C3CCC3)C2)=O)c(C)n[nH]c1C 35774,C(C(C(=O)N1CCOC2CC12)C(C)(C)C)NC(COC(CC)C)=O 35775,c1(C(=O)NC(C)CO)ccc2c(-c3cscc3C#N)nn(C)c2c1 35776,N1(C(C23CSCC2C3)=O)CC=CC(NC(C2(n3cnnn3)CC2)=O)C1 35777,C1(NC(C2N(C)CCC2)=O)CC2CC1N(C(=O)Cc1cccc(C3CC3)c1)C2 35778,Cn1cc(C(N2CC(NC(=O)CCOC3CC3)C(C3CC3)C2)=O)c(=O)n(C)c1=O 35779,C#CC1CN(C(=O)CCC2CCCCN2C(c2cc(Cl)no2)=O)CCO1 35780,C1(C(N(C2(CC(=O)NC(C#C)CC3CC3)CC2)C)=O)Cc2ccccc2C1 35781,C(=O)(C(C)(C)F)NC(C1CCCCC1)CNC(C(C)C1CCCC1)=O 35782,N1(C(c2cccc(CC)c2)C(=O)NCCCC2CC2)CCC(OC)C12CCCC2 35783,c1(C(C(N2CC(C(C)(C)O)(CNC(C(F)OC)=O)C2)=O)C)ccc(N(C)C)cc1 35784,C12(C(=O)NC(C(C)F)C)CC(CCO1)N(C(C1CN(C)C(=O)N1)=O)C2 35785,CCC(C)(C)C(=O)NCC1C2CN(C(=O)CNC(c3cccs3)=O)CC12 35786,c1(C(N2CC(NC(C3(CC)CC3(F)F)=O)C2)=O)ccccc1S(C)(=O)=O 35787,CCCC(C(=O)OC)NC(=O)CC1CN(C(=O)C=CCF)CC1C 35788,c1(C(=O)NCC2CN(C(C3CCC(=O)NC3)=O)CC2O)[nH]cc2c1CCC2 35789,N1(C(Cn2nnc(C)n2)=O)CC=C(C(=O)N2CCC(OC3CC3)CC2)CC1 35790,C(=O)(CCCCC(F)(F)F)NC12CC(NC(CC(C=C)C)=O)(C1)C2 35791,C(CC(C(C)(C)C)NC(c1c[nH]c(=N)c(C)c1)=O)N(C(C1C(CC)CCO1)=O)C 35792,CCCCCCC(c1nnnn1Cc1ccc(F)cc1)NCC(C)(CC)OC 35793,Cc1cnc(F)c(C(N2CCC(NC(c3cc(C(N)=O)ccn3)=O)C2C)=O)c1 35794,Cc1nnsc1C(=O)NC1(CNC(C2(C(C)C)CC2)=O)CC1 35795,CN1C(=O)OCC1C(=O)NC1CC(CNC(c2cccc(=O)o2)=O)C1 35796,c1(C(=O)NCCCN(C(C(C(=O)OC)OC)=O)C2CC2)cc2n(n1)CC(F)C2 35797,C12(C(=O)OC)CC1CN(C(=O)CC(O)CNC(c1cc(C3CC3)[nH]n1)=O)C2 35798,c1(C(N2C(C(N)=O)CCC(C)C2)=O)coc2c1CN(C(=O)CC1CCC1)C2 35799,C1(CC(=O)N(CCCN2CCCC(O)C2)C2CC2)CCC(F)(F)CC1 35800,N1(C(CC2CC(OC)C2)=O)CCC(CCNC(=O)CCc2cc(C)[nH]n2)CC1C 35801,c1(C(=O)NCC(CC)N(C)C(c2cnsc2C)=O)n[nH]c(C)n1 35802,C(=O)(C1=CCCCCC1)NCCN1CCN(C(c2cccc(N)n2)=O)CC1 35803,n1(C(C)C)ncc(C(N2CCCC2CN(C(=O)CSCc2ncc[nH]2)C)=O)c1N 35804,CC1=C(C(=O)C(=O)CCCCCC#N)COCC1.C1(CN)(C)CC1(F)F 35805,CCCC(C)CC(=O)NCC(O)CN(C(=O)COc1ccc(CC(N)=O)cc1)C 35806,N1(C(C=CC(=O)OCC)=O)CC2CC(NC(=O)Cc3cnco3)CC2C1 35807,C1(NC(c2cnsn2)=O)CN(C(C2CC(C(F)(F)F)C2)=O)CC1C1CC1 35808,N1(C(C)C)C(C)CN(c2cc(NC(c3nccs3)C)ncn2)CC1C 35809,Cc1ccc(C=CC(=O)NC2CC2NC(c2cnc(C(C)(C)C)s2)=O)cc1Cl 35810,c1(C2(C(=O)NCC(C)CN(C(=O)CO)C)CC2C(F)(F)F)ccccc1 35811,c1(OCC)ccc(NC(=O)CC2CC(NC(c3occc3COC)=O)C2)cn1 35812,N1(C(CC(CC)SC)=O)CC(NC(=O)Cc2cnn3ccccc23)C2(CCC2)C1 35813,C1(NC(C2C(CCOCC)C2)=O)CCC(CNC(=O)CC(C)(C)O)CC1 35814,C1(C)(OC)CCN(C(=O)C(O)CCCNC(=O)COc2ncccn2)CC1 35815,C1(C(N2CC(F)(C(=O)OC3CN(C(COC)=O)C3)C2)=O)CC(C2CC2)=NO1 35816,CC#CCC(C(=O)NCCC1(COC)CCN(C(C)=O)C1)NC(=O)OC(C)(C)C 35817,Cc1cc(F)cc(Br)c1C(=O)NC1CC2CCC1N2C(C1CCC(=O)C1)=O 35818,c1(C(=O)NC(CCC2CC2)C(=O)NCC(O)CCO)ccnc2cc[nH]c12 35819,c1(C(=O)Nc2cccc(C)c2C)cccc(S(=O)(=O)NC(C)CO)c1 35820,c1(-c2n(CCCOC)c(N3CCN(CC4CC4)CC3)nn2)c(C)c(C)n(C)c1C 35821,C#CC1(N(C)C)CCN(C(=O)OC2CN(C)C(C)(C(=O)NC(C)(C)C)C2)CC1 35822,c1(CN(C)CCOCCNC(c2cc(Cl)c[nH]2)=O)ccc([N+](=O)[O-])cc1 35823,C1(S(C)(=O)=O)(C(=O)NCC(C2CCC2)NC(CC=C(C)C)=O)CC1 35824,c1(C(C)C)nnc(C(=O)NCCC(C)N(C(=O)CC2CC2C)C)s1 35825,c1(C(=O)NC2CC(NC(C3CCCO3)=O)C2)c[nH]cc(F)c1=O 35826,N1(C(Cc2n(C)cnc2)=O)CCC2(CCC(NC(c3ccc(=O)oc3)=O)C2)CC1 35827,CC1(C)CCC(C(N2CC3CC3(CNC(c3ccc(Cl)o3)=O)C2)=O)O1 35828,N1(C(c2scc(C(C)=O)c2)=O)CC(O)CC1CNC(=O)COC1CCOC1 35829,c1(NCC(C(C(C)C)O)(C)C)cc(S(=O)(=O)NCc2ncsc2C)ccc1C#N 35830,CCC1=NOC(C(=O)NCCC(O)CNC(=O)C(F)(F)CO)C1 35831,CC1(F)CN(C(=O)C(O)C2CCC2)CCN(C(c2c(Cl)ccnc2F)=O)C1 35832,c1(CCNC(C(=O)OC=C)=O)ccc(C(N2CCCC2c2ccco2)=O)cc1 35833,N1(C(CSC)=O)CC2CC(C(=O)NCCC(O)CO)C(C2)C1 35834,C1(Nc2ncc(C(N3CCCC(C)(C(=O)NCC)C3)=O)s2)CCCCN(CC)C1 35835,CCCCCCCCCC(=O)NC1CN(C(c2cc(C(N)=O)c[nH]2)=O)CC1(C)C 35836,C(=O)(CCCCCNC(C1C(C)(C)C1(F)F)=O)NCc1nc(CC)sc1 35837,C12(C(=O)NCC(CN(C)C)O)CC(C)(CN1C(=O)CCc1ccccn1)C2 35838,C(=O)(C(CO)C(F)(F)F)NC(C(C)O)C(=O)NC1CC(C)(C)OC1=O 35839,C(=O)(C(F)C(F)(F)F)N(C)CCNC(C1CCC(Oc2ccncc2)C1)=O 35840,C1(C(=O)NCCCF)CCCCN(C(C2CCO2)=O)C1 35841,CC1CC(=O)NC(C(N2CC(NC(c3cn(CCC(C)(C)C)nn3)=O)C2)=O)C1 35842,c1(C(N2CCOCC(CC)C2)C(=O)NCCCCCC)ccn(C(C)C)c(=O)c1 35843,c1(C(N2C(CC)CN(C)CC2)=O)ccc(S(=O)(=O)N(CC(C)C(F)(F)F)C)cc1 35844,c1(CN=C(NC(C#C)C(C)(C)OC)NC2CCC2)ccc(C#N)cc1Cl 35845,CCC(C)C(C(=O)N(CC(C)(C)C(=O)NCC1=NOCC1)C)OC 35846,Cc1cc(C)c(C(=O)NC2CC23CC(NC(C2CCC(C)(C)O2)=O)C3)[nH]1 35847,C=C(CNC(=O)C(O)C1CCC1)CCNC(=O)Cc1cccnc1 35848,CCCCCC(CC)C(=O)NC(CNC(c1nocc1C)=O)CO 35849,c1(C(=O)NC(CNC(C(CC)n2nccc2C)=O)C2CC2)cc2cccnn2n1 35850,c1(C(=O)NC2C(NC(C(C)O)=O)COC2)cnc(C2CCC2)nc1O 35851,CCCC(C(=O)NC)NC(=O)CC1(N(C)C(C2CC(C)(C(N)=O)C2)=O)CC1 35852,N1(C(C(=O)NCC2CC2)=O)C(C(=O)NCCC2(O)CCC2)CC2CCCC12 35853,c1(C(=O)NC(CNC(c2cc(CC)n(C)n2)=O)C2CCC2)nccc(C#N)c1F 35854,C1(CC)CCCCN1C(=O)COCCNC(=O)CCC1CC1(C)C 35855,N1(C(C=CS(C)=O)=O)CC(NC(=O)Cc2cccc3c2CCC3)C(C2CC2)C1 35856,C(C(C)C(C)C(=O)NCC1(C(=O)NC2CCC(=O)N(C)C2)CC1)OC 35857,C1(CC(=O)OCC(C)(C)COCC(=O)Nc2ccccc2)C(F)(F)C12CC2 35858,CCC(Cc1ccccc1C)C(=O)N1CC(NC(c2csc(CO)n2)=O)C(C)C1 35859,C1(CC(C)NC(CCC2CC(C)C2)=O)CCN(C(c2nccn2C)=O)CC1 35860,c1(C(N2CCC(NCC3CCCOC3c3ncc[nH]3)C2)=O)cc(F)c(O)c(Cl)c1 35861,C1(CC=C)(NC(C2CCC(CC)CC2)=O)CCN(C(c2c[nH]c(Br)c2)=O)C1 35862,C1(C=O)(COC)CN(C(c2ccc(CO)o2)=O)C1.N(CC)CC1CC1 35863,N1(C(C2(C)N(C(Cc3c(C)ocn3)=O)CC=C2)=O)CCC(N=[N+]=[N-])C1 35864,N1(C(C(C)N=[N+]=[N-])=O)CC2CCCC2(CNC(c2cnnc(O)c2)=O)C1 35865,C(=O)(C(C)(C)CCCO)NCCC1CCN(C(C(C(C)(C)C)NC(N)=O)=O)CC1 35866,Cc1nocc1NC(=O)COC(=O)C(C)NC(c1ccc(F)s1)=O 35867,N1(C(CC2CC(=C)C2)=O)CCCC(O)(CN(C(=O)CCCn2cccn2)C)C1 35868,C1(C(=O)NC(C)CNC(C2CC(=O)N(c3nccs3)C2)=O)C2C3CCC(C3)C12 35869,N1(C(C2N(C(c3c(C#C)cn(C)n3)=O)CCC2(C)C)=O)CC2(COCC(=O)N2)C1 35870,N1(C(C(=O)N(C)CC2CCCN2)=O)CC2CCCC(N)C2C1 35871,c1(C(=O)NCC(C)(C)Nc2nc(COC)nc(Cl)c2)ccc2c(c1)nc(O)n2C 35872,c1(OC)cc(C(=O)NCC23CC2CN(C(c2n[nH]cc2C)=O)C3)nc(Br)c1 35873,C1(C)(CNC(CN(C)C(N)=O)=O)CN(C(=O)CC2CCCC23CC3)CCO1 35874,C1(CNC(CCC(C)OC)=O)CN(C(c2nnn(C(C)C)c2C)=O)CC(C)(C)C1 35875,N1(C(c2ccc(F)s2)=O)CC2CCN(C(c3nccc4[nH]ccc34)=O)C(C2)C1 35876,c1(OC)cccc(C(c2nnnn2CC(F)F)NCC2CC=CC2)c1OC 35877,c1(C(N2CCC(N(CCC)C(C3C=CCC3)=O)C2)=O)c(CC)nn2ccccc12 35878,c1(C(N2CCC(NC(Cc3c(C)occ3)=O)C(O)C2)=O)ccsc1S(N)(=O)=O 35879,N1(C(Cc2c(C)n(C)cn2)=O)CC(NC(C2(Cl)CC2(F)F)=O)CC(C)C1 35880,C1(C(=O)NC(C2(O)CCN(C(=O)CC3CC3)C2)C)C2CCC1(c1ccccn1)C2 35881,c1(CC)ccc(C(=O)NCC(CO)NC(c2ccc(C)cc2C)=O)cc1C#N 35882,n1(CC)cncc1CNCc1cc(C)on1 35883,c1(COC)c(C(=O)NC2CCNC(C(=O)O)C2)oc2ccccc12 35884,c1(C(N2CCC(N3CCN(C(CC)=O)CC3)CC2)=O)c(F)cc(F)cc1Br 35885,CC1CCCCC1C(=O)NCC(C)(C1CC1)NC(c1cnn(C2CC2)c1)=O 35886,CC(C)(CC1CCOC1)C(=O)NCC1CCN1C(=O)COCC1CCOCC1 35887,N1(C(CCC(C)SC)=O)CCC(NC(C2(C(F)(F)F)CC(F)(F)C2)=O)CC1C 35888,C1(NC(C2(OCC)CCSCC2)=O)COCCN(C(c2csnc2Cl)=O)C1 35889,N1(C(=O)CCc2cc[nH]n2)CCC2(CCCN2C(c2ccccc2Cl)=O)C1 35890,O=C(CC1=CCCCC1)NC1COCCN(C(c2cc3n(c2)CCC3)=O)C1 35891,N(C1=NC2CC3CC3C2(C)C1)Cc1ccc(OC(C(F)F)(F)F)nc1 35892,C(C(F)(F)CNC(=O)C(CC1CC1)NC(=O)CCOC(C)=O)OC.C(C(C)(C)C)O 35893,c1(C(=O)NC2CC(F)CN(C(C3CCCO3)=O)C2)nnn2c1CSCC2 35894,C(=O)(C1=CCS(=O)(=O)C1)N(C)CC1CCCN1C(=O)CC1CCCC(=O)N1 35895,C#CCC(CC(=O)NCc1cccc(C#C)c1)NC(c1cnn(C)c1Cl)=O 35896,c1(C(N2C(CNC(Cc3n(C)ncc3Cl)=O)CCCC2)=O)coc2c1COC2 35897,Cc1nn(CC(N2CCCC(C(C)NC(=O)Cn3nnc(=O)[nH]3)C2)=O)c(=O)o1 35898,C1(NC(C=C(CC)C)=O)CC2C=CC1N(C(=O)CCNC(=O)OC(C)(C)C)C2 35899,N1(C(C2CCC(C)O2)=O)CC(CNC(c2cc3ccccc3o2)=O)OC(C)(C)C1 35900,C1(NC(=O)CN(c2ccccc2)CCO)C2CN(C(=O)C(F)=C3CCC3)CC12 35901,N1(C(C(F)=CC)=O)CCC2(NC(c3cccc(Br)c3C)=O)CCCCC12 35902,c1(C(N2CCCC(C(=O)Nc3cnc(Cl)nc3)C2)=O)cnc2ccccn12 35903,N(C1CCc2cc(CNC(c3cn(C)nc3C)=O)ccc21)C(C(CCC#C)O)=O 35904,c1(C(=O)OC)ccc(C(=O)NC2CC3C=CC2C3)c(C(C)C)c1 35905,CC1(NC(c2nsnc2O)=O)CCN(C(C2CC3CC2C3)=O)C1 35906,C1(N(C(CSCCOC)=O)C)CC(CNC(=O)C(C)N(C(C)=O)C2CC2)C1 35907,C1(C(=O)NC2COCC2NC(c2cnc(O)s2)=O)(OC)CCOCC1 35908,Cc1cc2ccccc2cc1C(N1CC2CC(NC(=O)C3=COCCC3)C1C2)=O 35909,C(CC)(CC(=O)NCC1(CO)CCCC1)NC(CC=C)=O 35910,S(=O)(=O)(c1cccc(CNC(c2oc(C)nc2CN)=O)c1)N(CC)CC 35911,Cc1cc(F)ccc1C(=O)NC1CCCN(Cc2scnc2C)C1 35912,Cc1cc(C(=O)N(CCCCNC(c2ccc(CO)nc2)=O)C)c(Cl)cc1Cl 35913,N1(C(C(C)N(C)C(C2CC(=O)C2(C)C)=O)=O)CC2(CO)CC2(CO)C1 35914,C(CC(=O)NCCN(C)C(c1csnc1-c1ccccc1)=O)(C(C)C)OCC 35915,CC(=O)n1ccc(=NC(=O)N2CCC(c3ccccc3COC(C)(C)C)CC2)[nH]1 35916,c1(OCC)nccc(C(=O)NCCC2(NC(c3ccc(F)c(C)c3)=O)CC2)c1F 35917,c1(C(N2C(CNC(Cc3c(SC)cccc3)=O)C=CC2)=O)cccc2c1OCO2 35918,C(c1cc(Cl)c2c(c1)OCO2)=CC(=O)NCC(C)N(C)C(C1CCN(C)C1=O)=O 35919,c1(C(=O)NC(C)C(CO)NC(c2cnc3ccccn23)=O)cccc2nn[nH]c12 35920,c1(C(=O)NCCN(C(CCC#C)=O)CCC)cc(Br)c(OC(C)C)s1 35921,CCCCN=C(NCC1(O)CCC1)NCC1CCCCN1S(C)(=O)=O 35922,CC1CN(C(=O)CCCC2CCC2)CCC1NC(=O)CCc1cncc(Br)c1 35923,C(=O)(CC(C)COC(C1(CNC(=O)OC(C)(C)C)CC1(F)F)=O)OC 35924,C1(NC(c2cc(CC)sn2)=O)C=CCN(C(c2nonc2N)=O)C1 35925,c1(C(=O)NCCN(C(CCC(=C)Cl)=O)CC)cc(C(=O)OC)cc(C(F)(F)F)c1 35926,c1(OC)ccc(F)c(C(N2CCCC2Cc2cn(Cc3cscn3)nn2)=O)c1 35927,CCC(C)CC(C(=O)NC1CN(C(C23CCC(C2)C3)=O)C1)NC(=O)OC(C)(C)C 35928,CCC(C)(C)OCC(=O)N(CC(C)CNC(C1(CO)CC1)=O)C 35929,N1(C(CCCC(C)=O)=O)CCN(C(=O)CC2(O)CCCCCC2)C(C)C1C 35930,C1(NC(CCCC(N)=O)=O)CC2CC1CN(C(C1(c3cnccc3Cl)CC1)=O)C2 35931,N1(C(C2(CC)CCCC2O)=O)CC2CCC1CN2C(=O)CSc1c(C)cccc1C 35932,C1(NC(c2cc(SC)c(C)o2)=O)(CNC(c2nccn2C)=O)CCCCC1C 35933,C1(C2CCN(C(=O)CCOCC(F)F)CC2)(NC(CC2C(C)CCC2)=O)CC1 35934,CC1(CNC(C2CC(C(F)(F)F)C2)=O)CCN(C(C2(O)CC(F)(F)C2)=O)C1 35935,Cc1ncc2n1CCC(C(=O)NC1(CF)CCN(C(c3ccncc3Cl)=O)C1)C2 35936,C#CCCCCCC(=O)N1CCC2CN(C(=O)CSC(C)C)CC12 35937,CCCCC(C)CCC(=O)NCC1CCC(NC(=O)COCCOC)CC1 35938,c1(C(N2C3C(NC(C4CC(OCC)C4)=O)CC(C3)C2)=O)sc2ccccc2c1Cl 35939,c1(OC)cccc(C(N2CCCNC(=O)C2)C(=O)NC(c2ccccc2)C)c1Br 35940,c12ccc(cc1C#N)c(=O)[nH]2.N1(C(C)=O)CCC(O)C1C(N1CCOCC1C)=O 35941,C12(CNC(C=CC)=O)COCCN1CCN(C(C13CCC(CC1)OC3)=O)C2 35942,CSC1=C(C(=O)NCC2(CCNC(=O)C(n3ccnc3C)C)CC2)CCCC1 35943,N1(C(c2n(CC)ncc2)=O)CC(NC(c2cncc(Cl)c2)=O)C(O)C1 35944,N1(C(CCc2ncn(C)c2)=O)CC(NC(C2CC3CCC3C2)=O)C2(CC2)C1 35945,C1(C(=O)NCC=C2CCN(C(C3(SC)CCC3)=O)CC2)CNc2ccnn2C1 35946,C1(CC)CCN(C(C2CN(c3nncs3)C2)=O)C1CNC(C1COCCN1C)=O 35947,C1(NC(C=Cc2ccc(SC)s2)=O)CN(C(C2(CO)CCCCC2)=O)CC12CC2 35948,c1(C(C(=O)O)C2(C3CN(C(CC(F)(F)F)=O)C3)CC2)ncccn1 35949,C1(CNC(C(=O)NCCNC(C)=O)=O)C2CCCC1N(C(c1[nH]cnc1C)=O)C2 35950,c1(OC)ncnc(C(F)(F)F)c1-c1nc(C2CCC(F)(F)CC2)nn1C 35951,CCCCCCCCC(CO)NC(c1cc2nc(Br)sc2[nH]1)=O 35952,N1(C(C2(CC)COC2)=O)CCC2(CC1)CC2(CO)CNC(C1CCCO1)=O 35953,Cc1nc(C(=O)NC2CC(C)(NC(C3(C)CCN(C)C3=O)=O)C2)c2ccccn12 35954,Cc1c(C(=O)NC2(C3CCCN(C(=O)CC4CC4)C3)CC2)oc2ccc(F)cc12 35955,c1(-c2ccc(CNC(CC(C)C)=O)cn2)ccc2c(c1)OCCN2 35956,C1(OC)CC(CNC(=O)C(=O)Nc2cccc(F)c2)N(C(c2ccc[n+]([O-])c2)=O)C1 35957,c1(CC)cc(C(=O)N(CCCC(=O)NCCC2CC2C2CC2)C)ncn1 35958,c1(C(=O)NC2C(NC(c3cc(C)nc(C)c3)=O)COC2)cc2nccn2c(O)n1 35959,C1(C(=O)NC2CCN(C(Cn3c(C)nnn3)=O)C2)CCc2nc[nH]c2C1 35960,N1(C(C2(C)CC(C)C2)=O)CCCCC2(C1)CN(C(c1nncs1)=O)C2 35961,C1(NC(=O)CC2CC2C(F)(F)F)CCCCN(C(=O)C=Cc2ccccc2)C1 35962,CCCC(C(=O)NCC1(C)CCCN1C(=O)C(F)C(C)C)OCC 35963,C(C)(CCCCN(C)C)(c1nnnn1CCCSC)NC1(C)CC(=C)C1 35964,S(=O)(=O)(c1ccc(NCCCC(C)(C)C)c(F)c1)N1C(C(C)C)CC(O)C1 35965,CCCC(C)(O)CC(=O)NC1CCCN(C(c2cccc3cc[nH]c23)=O)CC1 35966,N1(C(C(C)=C2CC2)=O)C2CCC1C(C(=O)NC(c1ccns1)C)C2 35967,c1(OC)cc2ncc(NC(c3cccc(C4(C)CC4)c3)=O)c(Cl)c2cc1OC 35968,N1(C(C2(C)COC2)=O)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2)C2CC12 35969,N1(C(c2nc3c(s2)CC(C)CC3)C(=O)NC(CC)(C)C)CCC(C2CC(F)(F)C2)C1 35970,c1(C(=O)NCC(CN(C)C(c2ccnn2C(F)F)=O)O)coc2ccc(O)cc12 35971,CC(CCc1ccccc1)CC(=O)N1CCCC1CN(C(=O)CCCN(C)C)C 35972,Cc1[nH]nc(CNC(=O)C(c2cccs2)NC(=O)C=Cc2cncs2)c1C 35973,c1(CC)cc(C(N2CCC(CC(=O)N(CC(C)C#N)C)C2)=O)on1 35974,N1(C(C(C2CN(C(C(C)S(C)(=O)=O)=O)C2)O)=O)CC2CC(CO)C(C2)C1 35975,C1(COC)CN(C(c2cc(Br)c(C)cn2)=O)CCN1C(c1cnc(O)o1)=O 35976,c1(C(=O)NCCC2N(C(CSc3onc(C)n3)=O)CCC2)c(C)cccc1C 35977,Cc1c(C(=O)N(C)CCOCCNC(=O)C(C)C(C)C)cnn1C1CCOCC1 35978,Cc1ccc(C(N2CCN(C(=O)CC3(N(C)C)CCCC3)CC2)=O)c(Cl)c1 35979,C1(CNC(C2(C(CC)(F)F)CC2)=O)(NC(C2CC3C=CC2O3)=O)CC(F)(F)C1 35980,N1(C(c2ccc(COC)o2)C(=O)NCCC#N)CCOC(C2CC(F)(F)C2)C1 35981,C(=O)(C1CCCn2ccnc21)N(C1CCN(C(c2c[nH]c(=N)s2)=O)CC1)CCO 35982,n1(CC(N2CCN(C(C(=O)NC)C)CC2)=O)ccc2ncc(Br)cc12 35983,N1(C(CCC2C(C)(C)C2)=O)CCOC2(CCC(Nc3ncc(Br)cn3)CC2)C1 35984,N1(C(C)C)CCCC1CC(=O)N(C)CC1CCN(C(c2ccsn2)=O)C1 35985,C1(CN(C(CC(C)O)=O)C)COCCN1C(c1cncc(C(C)(F)F)c1)=O 35986,c1(C(=O)NCCC(CNC(C(CC)O)=O)(C)C)c(Br)ccc(OC)c1C 35987,[N-]=[N+]=NC1CN(C(C2OCCO2)=O)CC1NC(c1c[nH]nc1-c1ccc(Cl)s1)=O 35988,Cc1[nH]c(C)c(C(=O)NCC2CN(C(c3cn(C(F)F)cn3)=O)CC2O)c1C 35989,c1(CC)onc(C)c1C(N1CCCC(C(=O)NCCCCC(=O)NC)C1)=O 35990,Cc1ncc(Cl)c(C(=O)NC(C)CN(C(=O)C(c2cc(F)cc(F)c2)C)C)n1 35991,N1(C(C(C(CC)C)O)=O)CC(NC(C2OCC2(C)C)=O)CC(C)(C)C1 35992,c1(C(=O)NCCC(C)(C)NC(C(C)OC2CCOCC2)=O)ccc2c(c1)COC2 35993,c1(C(N2CCN(C)CC2CNC(C2CCS2(=O)=O)=O)=O)ncnc2c1ccn2C 35994,C1(CCC)(CO)CCN(C(=O)C(CNC(=O)C(C)(CO)OC)CC2CC2)C1 35995,c1(C(=O)OC)cc2c(N3CC(CNC(=O)COCC(F)F)CC3C)[nH]cnc-2n1 35996,c1(C(=O)NC(CNC(c2ccc(C)nc2O)=O)(C)CO)nccc2ccccc12 35997,C1(C(N2CCCC(=C)C2)=O)CC1C1CN(C(C2(C)CNC(=O)C2)=O)C1 35998,Cc1cc(F)ccc1CC(=O)NCC1CC2(CC2)CN1C(=O)C(C)CF 35999,O=C(C#CC1CCCOC1)NC1CCCC2CN(C(c3cncs3)=O)CC12 36000,CC(C)=C=CC(=O)NCCc1ccc(CNC(=O)CN2CCCC2)cc1 36001,C(C(C(=O)N1CC(C(N)=O)C1)C(C)C)NC(C1(CC(C)C)CC1)=O 36002,C1(CNC(=O)Cn2cnnc2)(NC(c2cc(Br)no2)=O)CCCC1 36003,C1(CC)CN(C(=O)CCN2CCCS2(=O)=O)CC1NC(=O)C#CC1CC1 36004,C1(C(=O)OC)CN(C(=O)CCCn2cc(CC3(O)CC(C(=O)O)C3)nn2)CC1F 36005,C1(Cn2cc(CC(C(=O)OC)C)nn2)CCCCN(C(C2(F)CC2)=O)C1 36006,CC(CC(=O)NC1C=CC(CNC(=O)CCc2cnn(C)c2)C1)c1cnn(C)c1 36007,c1(NC(c2cnc(Br)s2)=O)cc([N+](=O)[O-])c(Br)cc1OC(F)(F)F 36008,C#CCCCCCC(=O)NC(C)(C)CN1CCN(C(C2CSCN2C)=O)CC1 36009,Cc1nc(C(C)NC(C2CCN(C(c3c[nH]nc3C)=O)C2)=O)n[nH]1 36010,c1(C(=O)NCCCCNC(C2CCCN(C(CC)=O)C2)=O)cc(F)c(F)c(F)c1 36011,C1(C(N(C(CCC)Cc2ccccc2)C)=O)CC2CC(=O)C1O2 36012,C1(COCC)CCCN(C(=O)C(C2CCOC2)NC(=O)CC2CN(C)C2)C1 36013,C(=O)(CCCCC(C)(C)C)N1CCC(NC(COCc2ncc(C)o2)=O)C1(C)C 36014,Cc1nc(C2CCCCC2)nc(O)c1CCC(=O)N1CC(NC(=O)CO)C1 36015,c1(C(N2CCC(NC(c3c(C=C)cnn3C)=O)C2)=O)c(Cl)ccc(F)c1F 36016,N1(C(CCN(C)CC)=O)CCC(C)C1CNC(=O)Cc1ccc(C(F)F)cc1 36017,C1(O)(C(=O)NC2CCN(C(C3CC(C(=O)OC)C3)=O)C(C)C2)CCC(C)(C)CC1 36018,N1(C(C(CN(CC)CC)F)=O)CCC(F)(NC(=O)CC2CCOC2C)CC1 36019,C1(NC(C(=O)N(C)C)=O)CCCN(C(c2coc3c2COC3)=O)CC1 36020,n1(CCC(=O)NC(CNC(=O)CCC2CC2CC2CC2)C2CC2)ccccc1=O 36021,N1(C(C2CC(=C)C2)=O)C2CCC(C(=O)NC(C3CCCCC3)(C)C)C1CC2 36022,N1(C(CCCOC)=O)CC(F)(F)CC1CCNC(C1CC1(Cl)C(=O)OC)=O 36023,Cn1nc(C(=O)NC(C23CCC(CC2)C3)CNC(=O)Cc2ccco2)cc1Cl 36024,C1(NC(C(C)(CNC(CC=CC=C)=O)OC)=O)CC2(CCC2)C1OC 36025,c1(OC)cc(C(=O)NCCN(C(=O)CCCF)Cc2cccc(Cl)c2)cc(Cl)n1 36026,C1(C(=O)NCC2(OC)CC2)CCCCC1NC(=O)C(C)(C)C1CC1 36027,C1(C(=O)NC2CCC(NC(Cc3ccn(C(C)C)n3)=O)C2)CC2(CCO2)C1 36028,Cc1cccc2c1CC(C(N1CCC(NC(c3occc3Cl)=O)C1)=O)O2 36029,Cc1c(C(=O)NCCC(O)CNC(=O)CC(O)Cc2ccccc2)cccc1F 36030,c1(C(N2CC3(N(C(C4CC(CC)(CC)C4)=O)CC3)C2)=O)cnc2c(C)cccn12 36031,N1(CCn2c(C)ncc2)CCCC(C(=O)NCC2=CCCCC2)C1 36032,O=C(C1=C(Cl)CCCC1)NC1CCCC1C(N1CCC(c2nc[nH]n2)C1)=O 36033,N1(C(C(c2ccccc2)C)=O)CCCC1CCCNC(=O)CCc1cccnc1 36034,CN1CCC(C)(C(N2CCOCC2CN(C(=O)C(C)(C)c2ccns2)C)=O)C1=O 36035,C1(NC(c2cc(OC)ncc2)=O)CN(C(c2nc(C)ncc2Cl)=O)CC2(CC2)C1 36036,C(=O)(CCCC(F)(F)F)NCC1(NC(c2c(SC)cnnc2)=O)CCCCC1C 36037,c1(CC)cc(C(=O)NCC2CCCN(C(=O)CC3CC(F)C3)C2)cc(O)n1 36038,N1(C(C2(COC)CCCO2)=O)CCCN(C(c2cnn(C3CC3)c2C)=O)CCC1 36039,C1(CNC(=O)Cc2ccc(Cl)s2)CN(C(C2CC3(CCCO3)C2)=O)CC12CCC2 36040,N1(C(CCC=CC)=O)CCOC(C)C1C(=O)NCCC(C)C(C)C 36041,[N-]=[N+]=NC1COCC1NC(=O)Cn1cc(CON2CCC3CC23)nn1 36042,C1(CNC(CN(C(C)C)C(C2CC(=O)CS2)=O)=O)CC2(CCC2)C1 36043,n1(CC)cc([N+](=O)[O-])c(C(=O)NCC(O)CN(C(=O)CNC(=O)OC)C)n1 36044,N1(C(c2nc(O)cc(C(C)(C)C)n2)=O)CCC2CCC(C1)S2 36045,C1(C(=O)NC(CCC)C(=O)NCC2CCOC2C)CCCCC1(C)C 36046,Cc1ccnc2ccc(C(=O)NCC34CC3CN(C(C3CCC3(F)F)=O)C4)cc12 36047,N1(CC(=O)NC(CNC(C2CN(C(N(C)C)=O)C2)=O)C2CC2)CCCCC1 36048,C1(NC(C2CC(=C)C2)=O)(COC)CCCN(C(c2ccc(F)c(Cl)c2)=O)C1 36049,c1(CC)cc(C(N2CCC(C(C)NC(c3cn(C(C)C)cn3)=O)CC2)=O)nn1C 36050,C(=O)(C(C)C(F)F)NCCC1CC(NC(C(C2CCCC2)OCC)=O)C1 36051,CC(O)C(C(=O)N1CC(C2CCCO2)C1)NC(=O)COc1cccnc1 36052,c1(N(C)C)nccc(N(C2CC(N)C2)Cc2ncccc2C(=O)O)n1 36053,N1(C(c2n(CC#C)ccc2)=O)CC(NC(c2cc(CC)cc(F)c2)=O)C2CC2C1 36054,c1(C(=O)NCCCOCC(C)C)ccc(CNC(=O)Cn2cnnc2O)o1 36055,N1(C(Cc2ccc(C(C)=O)cc2)=O)CCC(CO)C(NC(c2cc(C)[nH]n2)=O)C1 36056,S(=O)(=O)(c1cccc(Cl)c1)N1CCC(C(=O)NCCOCCC)C1 36057,Cc1ccc(C)c(NC(C2(O)CCN(C(=O)Cc3cc(F)ccc3Cl)C2)=O)c1 36058,N1(C(C(C)C)=O)CC(C)(C)OCC1CNC(=O)C(C(C)C)n1cccc1 36059,C(=O)(C(F)C(C)(F)F)NC(CC(=O)N(C1C(C)COCC1)C)CC1CC1 36060,N1(C(Cn2ncc(C)c2)=O)CC2CC1CN2c1cc(-n2cncn2)ncn1 36061,c1(NC(C)=O)c[nH]c(C)c1C(=O)NC(C)CCNC(C1(F)CCOC1)=O 36062,N1(C(C(C(C)(C)C)(C)C)=O)CCCOC2CCCC12 36063,Cc1nn(C)c(N2CCOCC2)c1CNC(=O)NCC12CCN(CC1)C2.CCN 36064,C(=O)(C(CC1CC1)OC)NCC(CNC(C1(c2ccno2)CC1)=O)OC 36065,C(=O)(CC(C(F)F)NC(=O)Cc1ncn(C)c1C)N1C(COCC#C)CCC1 36066,c1(CNCCCNC(=O)Nc2cnc(N(C)C)nc2)ccc(F)c2ccccc12 36067,C(=O)(C(O)C(C)(C)C)NCC1(O)CN(C(C2(CC=C)CCC2)=O)C1 36068,Cc1cc(C2CCN(c3nnnn3Cc3cc(-c4ccco4)on3)C2)cc(C)c1 36069,C=CCC(C)(C)CC(=O)N(CCCOCCNC(c1c(C)coc1C(C)C)=O)C 36070,N1(C(C2C(CCOC)C2)=O)CC2(CC(NC(=O)C=CC(=O)N(C)C)CO2)C1 36071,n1(CCNCc2ccc(C(F)(F)F)s2)c(-c2cccs2)nnc1S 36072,C(c1c(Cl)nc2sccn12)=CC(N1CC(NC(C2CC3C=CC2O3)=O)C(O)C1)=O 36073,c1(C(=O)OCC)cccnc1N1CCC(NC(c2conc2CC)=O)CC1 36074,Cc1nc(O)nc(C)c1CC(N1CC=C(CNC(=O)CCCN(C)C)CC1)=O 36075,Cc1ccc(F)cc1C(N1CCC(C(F)F)(CNC(=O)Cn2cncn2)C1)=O 36076,CCCN=C(NCC1(C2CC2)CC1)NC1CCN(CC)C(C)C1 36077,CC1CCN(C(=O)CCn2cccc2)CC1NC(c1ccnc(OC(F)F)c1)=O 36078,Cc1cc(C(=O)NCC2(O)CCCN(C(=O)C=C(Cl)Cl)C2)c(C)n1C1CCOC1 36079,c1(-n2c(COC(F)F)nc(C(C)SC)n2)cccc2nc[nH]c12 36080,C12(NC(c3n(C=C)nnc3)=O)CCN(C(c3c(Cl)cnn3CC)=O)CC1C2 36081,c1(C(N2CC(NC(C3CN(C)C(=O)C3)=O)C(O)CC2)=O)nccn2nccc12 36082,c1(C(=O)NCC2CCCN(C(C3CC(C)C3)=O)CC2)cn(C)c(=O)nc1O 36083,C(CCCCC(=O)N1CCOCC(CNC(C2CC23CC3)=O)C1)OCC 36084,C1(NC(C(CC)N(C)C)=O)CCCCC1C(=O)OC.C123CC(C1)(C2)CNC3=O 36085,C1(C(=O)NCC(CNC(CC2CCC(=O)C2)=O)O)CC2(CCOCC2)C1 36086,C1(N(C(=O)C(F)Cc2ccccc2)C)CCCN(C(=O)OC(C)(C)C)CC1 36087,C1(C(=O)NC2CC2C2CCCN(C(C3CC34CC4)=O)C2)CCCCC12OCCO2 36088,C1(NC(C2C(C)=CCS2)=O)CN(C(c2csc(C)n2)=O)CC1(C)C 36089,C12(CNC(C3CC(=C4CCC4)C3)=O)CCC(C1)N(C(=O)COc1ccsc1)C2 36090,N1(C(C(C)c2cccs2)=O)CCC2(CCN(C(c3cnn(C)n3)=O)CC2)C1 36091,c1(SCC#N)cccc(C(=O)NCC(O)CNC(=O)CCN2CCCC2)c1 36092,Cc1cc(CN2CCOCC2C(=O)Nc2cnc(I)c(Cl)n2)ccc1O 36093,CCCCC(F)C(=O)NCC1C(C(N2CCCC(OCC3CC3)C2)=O)C1(C)C 36094,c1(C(=O)NC2CCCN(C(c3ccc(CO)o3)=O)CC2)cn2c(Cl)cccc2n1 36095,c1(C(=O)OCC)cnc(SC)nc1N1CCC(O)C1C(N1CCCC1)=O 36096,C1(NC(CCOC)=O)CC2CCC(C1)N2C(c1cnc(O)c2ccsc12)=O 36097,N1(C(c2c(C)nc(=N)[nH]c2C)=O)CCC2CCN(C(c3ccoc3Br)=O)CC2C1 36098,CC1C(NC(C2C=CCC2)=O)CCN1C(=O)Cc1cn(C)nc1Cl 36099,C=CC(C)(CC)C(=O)NCC1CC1CNC(c1nc(N(C)C)nc(=N)[nH]1)=O 36100,C(=O)(CCCc1cccnc1)NC(CN(C(c1cnccn1)=O)CC)C 36101,N1(CC(=O)NC23CC(CNC(Cc4c(C)n[nH]c4)=O)(C2)C3)C(=O)C(C)C(C)C1=O 36102,c1(C(N2C(CNC(C3CC3C3CCCCC3)=O)CCC2)=O)nc2cnccc2s1 36103,c1(CC)nn(C)cc1C(=O)NC1CCN(C(=O)Cc2cnc[nH]2)C1C(C)C 36104,C12(NC(c3c(C)ccs3)=O)CCCN(C(C3(CS(C)(=O)=O)COC3)=O)CC1C2 36105,C1(C(=O)NCc2c(C(=O)NCCC(COC)O)nco2)OCCCC1(C)C 36106,CCCCC(O)C(=O)NCC1(C)CCN(C(c2ncccc2C2CC2)=O)C1 36107,N1(C(C=CC(C)N(C(Cc2c(C)scc2)=O)C2CC2)=O)CCOC2CCCC12 36108,C(=O)(CN=c1[nH]c(C)cs1)N1CCC(CNC(c2c(OC)nccc2)=O)C1(C)C 36109,C1(C(=O)OC)CC(C)(C)CN1C(CCC1CCCC1)C(=O)NC1CCCC1 36110,C(CCCCOCc1cc(C(=O)OC)no1)NC 36111,c1(C(=O)NC(CCNC(c2c(CC)nns2)=O)C)cc(Cl)ccc1OC 36112,c1(C(=O)NCC(C2CCCCCC2)NC(CCOCC#C)=O)nnc(O)cc1O 36113,N1(C(CSC)=O)CC2CC3CC2C1C3NC(=O)CCc1ccc([N+](=O)[O-])cc1Cl 36114,Cc1snnc1C(=O)NCCOC1CCN(C(c2cnn(-c3nccs3)c2)=O)C1 36115,C1(NC(CN(C)CC)=O)(CC)CN(C(=O)CC(C)c2ccccc2)C1 36116,CCC(C)(COC)C(=O)NC1CN(C(c2cccc(F)c2C)=O)CC1F 36117,CC1Oc2ccc(CNC(=O)NC3(C)CCC(=O)NC3=O)cc2N(C)C1=O 36118,N1(C(C2=C(C)CC2)=O)CCC2CN(C(c3cc([N+](=O)[O-])ccn3)=O)CC12 36119,c1(C(=O)NCc2ncoc2CCNC(C2(CCF)CCC2)=O)ccnc(S)c1 36120,c1(OC)ccc(Cl)c(C(=O)NC(C)CCNC(C2CC(C3CCC3)C2)=O)c1 36121,c1(C(=O)NCC2CC(NC(c3ncccc3F)=O)C2)cc2c(nc1O)CCCC2 36122,c1(C(C)C(N2CCCC2C(C)(C)NC(c2cnoc2)=O)=O)ccc(F)cc1 36123,c1(N(C)CC2C(C)C2)ccc(S(=O)(=O)N2CCCN(C)CC2)cc1Cl 36124,N1(C(CSCC)=O)CCC(NC(c2ccc3c(c2)CCO3)=O)C(F)(F)CC1 36125,n1(CC)ncc(C(=O)NCCn2cc(CNC(c3c[nH]c(=N)s3)=O)nn2)n1 36126,CCC(C)CC(C)N(C(=O)CCNC(c1cn(C)cc1C)=O)C 36127,c1(C(=O)NCC2C(C)CN(C(c3csc(Cl)c3)=O)CC2)cc2ccsc2c(O)n1 36128,c1(C(=O)NCC2CC(C)CN(C(=O)CCCC(C)(C)C)C2)nn(C)cc1[N+](=O)[O-] 36129,N1(C(=O)Cn2ncnn2)CCCC1C1(C(=O)NCCn2cncn2)CC1 36130,c1(C(C(=O)OCC(N2CCN(CC)C(=O)C2)=O)N(C)C)ccc2n[nH]cc2c1 36131,C1(NC(c2n(CC)ccc2)=O)C2CC3C(C2)C13C(=O)NCC(C)OC 36132,c1(C(=O)NCC(CN(C(C2CCN(CC(C)C)C2)=O)C)C)cc(S(N)(=O)=O)co1 36133,C(=O)(CC(C)C(F)F)NCC(CC)(C)NC(=O)Cc1nc[nH]n1 36134,CC1(C)CCC(C(=O)NC2CCc3n[nH]cc3C2)CN1C(=O)CC1CCSC1 36135,Cc1ccc(F)c(C(=O)NCCC(O)CNC(c2cc(C)n(C(C)C)n2)=O)c1F 36136,C1(CC(=O)OC2(c3c(OC)ccc(F)c3)CC2)CC(O)C12CC(F)(F)C2 36137,CC(CC(=O)NCC(=O)NCC1CCN(Cc2ccc(Cl)s2)C1)c1cccnc1 36138,C=C(Cl)CCC(=O)N1CCC(C(C)(O)CNC(c2ccn(CCOC)n2)=O)CC1 36139,C(=O)(C(CC)CC(F)(F)F)N1CCCC(NC(CS(CCC)(=O)=O)=O)C1CC 36140,O(C1CCCc2ccccc21)CC(=O)N(CCCNC(C1CCO1)=O)C 36141,Fc1cc(NCCNc2nccc(SC3CCCC3)n2)cc(C(F)(F)F)c1 36142,c1(N(C(C)C(=O)N(C)CCCN)S(C)(=O)=O)ccc(F)cc1 36143,C1(C(=O)NC2CC(C)OC2=O)CN(C(C2CCC(O)C2)=O)CC(C)(C)C1 36144,N1(C(C2CCC(CCC)CC2)=O)CCCC2CN(C(=O)Cc3ccsn3)CCC12 36145,c1(OCCC(N2CCC(C(=O)NCC3(n4ccnc4)CC3)C2)=O)ccccc1 36146,C1(NC(c2cc(OC)ncc2)=O)CC2CN(C(C3CCOC3)=O)CC2C1 36147,C1(C)(CNC(Cc2nnc(C)o2)=O)CCCN(C(=O)CC2COC3CC2C3)C1 36148,c1(CC(=O)N(C)CC2(CNC(C3C=CC(C(=O)OC)C3)=O)CC2)ccc(Cl)cn1 36149,CC(C)=C=CC(=O)NC(C(=O)NOCC1CCCC1)C1CC=CCC1 36150,C12(CNC(c3n(COC)ncc3)=O)CCC(NC(c3cn[nH]c3)=O)(CO1)C2 36151,N1(C(C=CCOC)=O)CC2CCC1C(CNC(=O)C(CO)NC(=O)C(F)(F)F)C2 36152,N1(CC(=O)NC(c2ccc(-c3ccc(Cl)cc3Cl)nc2)C)CCc2[nH]nc(O)c2C1 36153,c1(C(=O)NC(CN(C(c2ccn(C3CCC3)n2)=O)CC)C)nc(C)sc1C 36154,C1(CC(=O)NCC(CC)NC(c2cnc(S)n2C(F)F)=O)C=NN(C)C1=O 36155,c1(C(N2CCC(O)(CNC(=O)C3=CCCC3)C2)=O)cccc(S(=O)(=O)C2CC2)c1 36156,C12(NC(CCc3n(C)cnc3)=O)CN(C(c3cccs3)=O)CC1CS(=O)(=O)C2 36157,Cc1cc(C)c(C(=O)NCC2(O)CC(NC(=O)Cn3ccnc3C(C)C)C2)o1 36158,C1(NC(CCOCCOCC)=O)CC2CC1CN(C(C1CC13CC3)=O)C2 36159,c1(C(=O)NC(CN(C(=O)CC2CCCC2)CC)C)cc(F)cc(Cl)c1 36160,CCC(C(=O)NC(CC1CCC1)C(=O)NC1CCOCC1O)C(F)(F)F 36161,C1(CCNC(C2(CC)CC2)=O)CN(C(c2c(NC(C)=O)nn(C)c2)=O)CCO1 36162,N1(CCNC(CCCOC)=O)CCN(C(c2ccc(C(N)=O)s2)=O)CC1 36163,C(C1CCN(C(=O)CCCN=[N+]=[N-])CC1)=CC(=O)NCc1nc(C(C)C)on1 36164,N1(C(c2cc(Br)co2)=O)CC2CCCC(C1)N2C(c1conc1C1CC1)=O 36165,C1(C(=O)NCC(C)(C)OCCNC(C2CC2Cl)=O)Cc2ccccc2C1 36166,C1(NC(C(CN(C(=O)CS(=O)CC)CC)N(C)C)=O)COCC(C)(C)C1 36167,Cn1ncc2c(N3CCCN(CC(F)(F)F)CC3)nc(=NCC(Cl)=CCl)[nH]c12 36168,c1(C(=O)NC2C(NC(C(C(C)C)N(CC)CC)=O)CC2)c(F)cccc1Cl 36169,n1(CCC(=O)N(CCCNC(=O)CSC(F)F)C)sc2ccccc2c1=O 36170,CN1CC2(CCN(C(c3cccc(C(F)F)c3)C(=O)NCC3CC3)C2)CC1=O 36171,N1(C(CSCC=C)=O)CCC2(CC(C(=O)NC3CC4CC3C(O)C4O)C2)C1 36172,C1(CNC(C(=O)NCC)=O)C2CCC(C2)N1C(=O)C(C)(C)C1CCCCC1 36173,C1(NC(c2cnn(C3CC3)c2)=O)CC2CN(C(=O)C3=COCCO3)CC2C1 36174,N1(C(c2c(N)cn(C)n2)=O)CC(NC(c2cc(CCCO)on2)=O)CC2(CC2)C1 36175,N1(C(COC2CN(C(C)=O)C2)=O)CCC(NC(c2nnc(C)s2)=O)CC(C)(C)C1 36176,C1(C(N(C2CN(C(c3ncoc3-c3cccs3)=O)C2)C)=O)C2CS(=O)(=O)CC12 36177,N1(C(c2cccc(OC(F)F)n2)=O)CC2CCC(C1)N2CC1CCCO1 36178,c1(NC(C(C2(O)CCC2)NC(CCN(CC)CC)=O)=O)cc(C#N)ccc1C 36179,c1(SC)ccc([N+](=O)[O-])c(C(=O)NC2CC(CCNC(=O)CC(C)C(C)C)C2)c1 36180,C(=O)(CCC(=O)N1CCCCC1C(C)NC(C1CN(CC(C)C)C1)=O)NCCC 36181,C1(NC(C2=C(C)CC2)=O)CCN(C(c2cccc(I)c2F)=O)CC1F 36182,C1(COC(c2ccn(CC(F)(F)F)n2)=O)CCCCN1Cc1nn[nH]n1 36183,C1(NC(CSC(C)C)=O)CC2(CCN(C(c3csc(C4CC4)c3)=O)CC2)C1 36184,CN1C2CCC1CN(C(C1COCCN1C(c1ccc(O)c(C#N)c1)=O)=O)C2 36185,Cc1cc(CC(=O)NCC2C=CC(NC(c3nccn3C)=O)C2)n(C)n1 36186,C1(C(=O)NCc2ccc(C)c(C)c2)N(C(=O)CC=C(Cl)Cl)CC12CCCC2 36187,Cn1ncc(Cl)c1C(=O)NCC1C=CCN1C(=O)Cn1ccccc1=O 36188,C1(C(=O)NC2CC(C3CNC3)C2)CNc2ccnn2C1 36189,c1(CCC)ccc(C(=O)NC2CC(F)(CNC(C3(C)CCC(=O)N3)=O)C2)cc1 36190,c1(OC)cc(CC(N2CCC(C)(NC(c3cc(C(C)C)on3)=O)C2)=O)cc(Cl)c1 36191,N1(C(CCCCOC)=O)CC2(CCCCN2C(C2(C)CC3CCC2O3)=O)C1 36192,N(C1CCCn2cnnc21)C(=O)Nc1ccc(C2CCC2)nc1 36193,Cc1ccc(C(=O)NC2CC(CNC(=O)CNC(c3cccs3)=O)C2(C)C)n1C 36194,Cc1ccc(S(=O)(=O)N2CC(C)NC(C)C2)cc1NC(=O)C(N)C1(C(C)C)CC1 36195,c1(CC(=O)NC2C(NC(C(C=C)O)=O)CCCC2)nn(C)c2ccccc12 36196,C1(OCCNC(=O)Cc2ccon2)CCN(C(=O)CCC2CC2(Cl)Cl)C1 36197,C(=O)(CC(CNC(=O)CN1CCC(=O)CC1)C1CCC1)N(C1CCN(C)C1)CC 36198,C(=O)(CC(c1ccccc1)C1CC1)NC1C(NC(C(=O)NCC(F)(F)F)=O)CC1 36199,c1(CCC(N2CCC(NC(C3(F)C(C)C3)=O)C23CC3)=O)ccc([N+](=O)[O-])cc1 36200,C(=O)(CCS(=O)(=O)c1ccccc1)NC(CC)CN(C(=O)C(C)CC1CC1)CC 36201,CCCC(CC)CC(=O)NCC12CC(CN1C(c1cccc(C#N)c1)=O)C2 36202,O=C(C1CCc2c[nH]nc21)NC1(C(N2CCn3nccc32)=O)CCC1 36203,C(=O)(CCCC(=O)N1CCC1(C)CC(=O)NOCc1ccc(O)cc1)OC 36204,C(=O)(CCCCN=[N+]=[N-])NCC(CN(C(C1(C2(C)CC2)CC1)=O)CC)(C)C 36205,Cc1cnc(CCNC(=O)CNC(C2(N(C)C)CC2)=O)nc1 36206,N1(C(C2N(C(C=C(COCC)C)=O)CCOC2)=O)CC(C2CC2)(CC)C1 36207,N1(C(c2ccc(C)c(F)c2)=O)CCCCCC(NC(C2(C)CC2(F)F)=O)C1 36208,C#CCCC(CCc1ccccc1)OC(c1ccc(Br)c(O)c1)=O 36209,N1(C(CCC2(NC(c3occ(C)c3)=O)CCCC2)=O)Cc2cccc(C)c2C1 36210,Nc1ncc(C(=O)NC2CC(NC(c3ccccn3)=O)C2)cc1-c1ccccc1 36211,c1(C(N2C(CN(C)C(c3scc(Cl)c3Cl)=O)CCC2)=O)cccc(=O)n1C 36212,CCCC(C(=O)NCCC(Cc1cn(CCSC)nn1)SC)c1cccc(Cl)c1 36213,N1(C(CCC(=O)N(C(C)C)C)=O)CCN(C(c2coc(C(F)(F)F)c2)=O)C(C)C1 36214,C1(C(=O)NC23CC(NC(Cc4c(N)ccc(Cl)n4)=O)(C2)C3)CCc2nccn2C1 36215,Cc1cc(C(N2C(C(N3CC(O)(c4nn[nH]n4)C3)=O)CC2C)=O)c[nH]c1=N 36216,C(=O)(C1CCCn2ccnc21)N1CCC(CNC(c2ccc(O)cc2F)=O)CC1 36217,N1(C(C)C)CC(NC(=O)CCCN(C(=O)CC2CSCCO2)C)C(C)C1 36218,c1(NC(CN2C(C)CC2)=O)cccc(NC(=O)Cn2ncc(Br)n2)c1 36219,C1(NC(C2CC(F)C(=O)N2)=O)CCN(CCNC(=O)CN2CCOCC2)CC1 36220,CC1CC=C(C(=O)N2CCCC(CCC(=O)NC3(C)CCCCC3)C2)CC1 36221,c1(C(=O)OC)ccc(C(=O)NC2CN(C(=O)C(N)=O)CC2OC)c(C)c1 36222,N1(C(C(CC(=O)OC)C)=O)CC2(CCCC2)C1C(=O)NCCC1(O)CCCCC1 36223,C1(CCCC)CCN(C(c2cc(CCNC(=O)C(C)Cn3cccn3)on2)=O)C1 36224,C=CCC(F)(F)CN(C(=O)C(C1CCN(C(=O)C(C)C2CC2)CC1)C)C 36225,c1(C(=O)NCCOCCCN(C(C2(CC)CC2)=O)C)cc2c(cc1Cl)CCCC2 36226,c1(C(=O)NC2(COC)CCN(C(C3CCCN3C)=O)C2)cn(C)c(=O)cc1OC 36227,Cc1ccc2c(c1)CC(N(C(=O)COc1nc(C(C)OC(C)C)no1)C)C2 36228,C1(CNC(c2ccc(N3CCC3)nc2)=O)CN(C(c2nccnc2Cl)=O)CCO1 36229,N1(C(C)=O)CC(C)OC2(CCN(C(c3c(C)nc(C(C)(C)C)nc3S)=O)CC2)C1 36230,c1(CC)nc(C)c(C(=O)N(C)CCOCCN(C)C(c2nc(C3CC3)cs2)=O)s1 36231,C12(CNC(CSCC=C)=O)CCC(CN1C(c1ccc(C)nc1OC)=O)C2 36232,c1(C(=O)N(c2cccc(Br)c2)CCO)cnc2n1CCN(C(c1occc1Br)=O)C2 36233,C1(CNC(c2ccnc(CO)c2)=O)CC2CC2N1C(=O)COCC1CCOCC1 36234,C1(NC(c2cnc(OC)s2)=O)CCCN(C(=O)Cc2cccc(F)c2F)C1C 36235,c1(C(C)NC(C2CN(C)C2)=O)ccc(CNC(c2ccc(C#N)[nH]2)=O)cc1 36236,N1(C(=O)NCCCCl)CCC2(CCCN(Cc3cccnc3F)C2)CC1 36237,N1(C(C2(CC=C)CCC2)=O)CC(CNC(=O)C(n2cc(C)cn2)C)C(O)C1 36238,c1(C(=O)NC2C(CNC(c3ncc(Cl)s3)=O)CCCC2)cnn2c1C(=O)NCC2 36239,C1(C(=O)NCc2ccc(C(=O)NC3CC(=C)C3)s2)CC(C)(C)CN1C 36240,C(=O)(CCCCC#N)N(CCC(C)NC(=O)CC1CCC(F)(F)C1)C 36241,C1(CNC(CCS(C)=O)=O)CCCC2(CCN(C(c3ncccc3Cl)=O)CC2)O1 36242,c1(C(=O)NCC(CN(C)C(C2CN(C3CCCCC3)C2)=O)O)cc(F)ccc1O 36243,N1(C(C(C)OCCC=C)=O)CC(NC(=O)CCn2cc(C)cn2)C(C)C1 36244,n1(CC#C)cccc1C(=O)NC(C)CNC(c1cc(C2CCC2)no1)=O 36245,c1(CC(=O)NCCC(C)NC(CC(CC)OC)=O)cccc(F)c1F 36246,c1(OC)ccc(F)c(C(=O)NCC2CC3(CC3)CN2C(=O)CC2CNC(=O)C2)c1 36247,C1(NC(C(CC)CC(C)C)=O)CCCC12CCN(C(=O)CC1CC(F)(F)C1)CC2 36248,N1(C(c2c(C)[nH]cc2)=O)CCC(CO)C(NC(=O)Cc2cn(C)cn2)C1 36249,C(=O)(C(O)CCSC)NC1(CCC(=O)NCCCC=CC)CCCC1 36250,C=CC1CN(C(=O)CC(C)CF)CC1NC(c1ccc(OC)cn1)=O 36251,C1(c2n(C)ncc2)CN(C(=O)C(NC2=NCCS2)=O)CCO1.C(CCC1CC1C)N 36252,C=C(Cl)C(C)(C)C(=O)N1CCCC(N(C)C(c2csc(C(C)(F)F)n2)=O)C1 36253,N1(C(C2CSCCS2)=O)CC2CCN(C(C3(O)CCSCC3)=O)CC12 36254,N1(C(C(C)(C2CC2)OC)=O)CCN(C(C23CC2COC3(C)C)=O)CC(O)C1 36255,N1(C(C(c2ccccc2)C)=O)CC(NC(c2c[nH]c(=O)cn2)=O)C(C)C1 36256,N1(C(C=CC2N(C)CCC2)=O)CCC12CN(C(C1(Cl)CC3CCC1O3)=O)C2 36257,CCCCCC(C)(C)C(=O)NCCC(C)NC(=O)C(n1cc([N+](=O)[O-])cn1)(C)C 36258,C(CCCCCCCO)=CC(=O)N(C1CN(C(=O)CCCCCC#N)C1)CC 36259,C#CCC(CC(=O)NC1CC2(NC(c3cn(C)nn3)=O)COC1C2)c1ccccc1 36260,C(=O)(CC(C)C(C)C)NCCC1(NC(c2cn(CCC=C)nn2)=O)CCOCC1 36261,c1(C(N2CC=CC(NC(C=CCN(C)CC)=O)C2)=O)cc[nH]c2nccc1-2 36262,C(c1cccc(C)c1)=Nc1ccccc1Cl.C12CC(C1n1cccn1)NC(=O)C(C)O2 36263,C1(C(=O)Nc2cccc(NC(c3cnn(C)n3)=O)c2)CC2(C1)CC2(F)F 36264,C1(C(=O)NC2(COC)CC2)CC12CC(NC(=O)CCC1CCCO1)C2 36265,c1(OCC)ccccc1OCCN1CC2C(C(=O)NC(CC)CO)C2C1 36266,C1(CNC(=O)COC2CCCC2)C(C2CC2)CCN1C(C12CCC(F)(CC1)C2)=O 36267,C(CC(CC)C(=O)NC(c1cnn(C)c1)C(=O)NC(COCC)C(C)C)=CC 36268,Cc1ccc(-n2nnc(CC(=O)NCC3COCC3N3CCOCC3)c2C)cc1 36269,O(NC(=O)C(O)CNC(=O)C(O)C(F)(F)F)C(C=C)C 36270,n1(CC(=O)NCC(CC)N(C)C(c2cnc(C3CC3)s2)=O)nnc(C2CC2)n1 36271,c1(C(=O)NC2CC3(CC(NC(C4C(C(=O)OC)C4)=O)C3)C2)ccnc2[nH]cnc12 36272,N1(C(C2(C(=O)OC)C(=C)CC2)=O)CCCCC(N(C)C(c2nn(C)cc2Cl)=O)C1 36273,C(=O)(C1CCCc2ncc(C)n21)N1CCC(NC(CCc2nnc(CC)o2)=O)C1 36274,c1(OC)ccc(C(=O)C(=O)NC2CCC(NC(=O)C=C(C)C)C2)cc1OC 36275,CC1CC(F)(F)CN1C(=O)C=CC(C)(C)NC(=O)C=CC1CCC1 36276,CCCC(C(=O)OC)C(=O)N1CCC(C)(C(=O)NC(c2cncnc2)C)C1 36277,C(C1CCOCC1)=CC(=O)NC1CC(NC(C2(C(N)=O)CCC2)=O)C1 36278,c1(C(=O)NCC2(F)CC(NC(CC(CN(C)C)O)=O)C2)ncnc2sccc12 36279,C=C=CC(C)C(=O)NC1(C)CC(NC(=O)CCc2nc(-c3ccoc3)no2)C1 36280,C(=O)(C(C)(C)CC#N)NC1C(NC(c2c(SC)cn(C)n2)=O)COCC1 36281,N1(C(C(C)CSC(F)(F)F)=O)CCCC(CNC(=O)Cc2nn(C)cc2Cl)C1 36282,c1(C(=O)NC(C(C)NC(CNS(CC)(=O)=O)=O)C)cc2oc(C)c(C)c2[nH]1 36283,c1(OC(C)C)ccccc1C(=O)N(C)Cc1cnc(C(F)(F)F)[nH]1 36284,C1(C(=O)NCCC2OCCN(C(C3C=C(C)CS3)=O)C2)CCCC(=O)N1C 36285,c1(C(=O)OCCCC#C)nnc(C(F)F)s1 36286,C1(C(=O)NC2CCC(NC(=O)Cc3ccccc3F)CC2)(COC)CCOCC1 36287,C=CC(CCC)CC(=O)NCC1CCN1C(c1cc(F)c(N)c(F)c1)=O 36288,N1(C(c2cc(C)[nH]c2)=O)CC2(C(=O)NC3CC4(C3)CC(C)C4)CCC1CC2 36289,C1(C(=O)NCC2(CC(=O)NCC)CC2)CCCCC1O.C1CC1OC(C)=O 36290,N1(C(CC(C)NC(=O)CSC(F)F)=O)CCCCC1NC(=O)CC(C)(C)C 36291,C1(C(=O)NCC2(NC(c3ccc(C)o3)=O)CC(OC)C2)CC12CCCCC2 36292,c1(C(=O)NCC2N(C(c3cc(COC)no3)=O)CC2)ccc([N+](=O)[O-])cn1 36293,CCC(CNC(C1(NC(=O)CCn2cncn2)CC1)=O)CCO 36294,Cc1ccc(C(=O)NCC2(F)CCN(C(=O)CC3CC=CCC3)CC2)c(O)n1 36295,N1(C(C(F)OC)=O)CC(NC(C2(CCF)CCOCC2)=O)C(C(F)(F)F)C1 36296,C(=O)(C(COC)CC(C)C)NC1(CC=C)CN(C(=O)C(C)=CC(C)(C)C)C1 36297,C12(C(=O)NCC3(C)OCCN(C(Cc4nnc(C)o4)=O)C3)CCCCC1C2(F)F 36298,Cc1ncnc(C(=O)N(C(CC(C)C)C(=O)NCc2csnc2C)C)c1C 36299,C1(NCc2ccccc2Cl)CCCN(c2ncccn2)C1.C12(CC1)N(C)C2 36300,c1(CC(=O)NC(CNC(C(C)OC)=O)(C)C)c(Br)ccc(Cl)c1F 36301,C(C)(C)(CC(=O)N(CC(O)CN(C)C(c1c(C)coc1C(C)C)=O)C)SC 36302,c1(C(N2CC(CNC(c3[nH]nnc3C3CC3)=O)C2)=O)cc2c(F)cc(F)cc2[nH]1 36303,c1(C(=O)NC2CC(CNC(C(CC)n3cncn3)=O)C2)cc(C)nc(O)n1 36304,C1(CC(=O)NCC(C2CCN(C(=O)C=Cc3cc[nH]n3)CC2)C)CCCCN1C 36305,C(=O)(C1COc2ccccc21)NCCN(C(CSCCC)=O)CCOC 36306,CC1CCC(CNC(c2coc(CNC(C3(C)CSC3)=O)c2)=O)N1C 36307,c1(C(=O)NC2CC(NC(C3N(S(C)(=O)=O)CC3)=O)C2)cc2nc[nH]c2cc1N 36308,N1(Cc2cn(C(C)C(=O)NCC3(n4ccnn4)CC3)nn2)CCN(C)CC1 36309,CC1(C(=O)NCCCCCNC(=O)CNC(c2ccncc2)=O)CCC(=O)NC1 36310,C1(NC(CSCCC)=O)CC(C)CN(C(c2c[nH]nc2Br)=O)C1 36311,c1(CNC(C2CC(C)CN(C(=O)CCC(=O)NN(C)C)C2)=O)ccc(C#N)cc1 36312,c1(C(=O)Nc2c(C(=O)OC)scc2)ccccc1N1CCNC1=O 36313,C=C=CC(C)C(=O)NC(CNC(c1cc(C)n(CC(F)(F)F)n1)=O)CC=C 36314,n1(CCC(=O)NCC2CC(OC)CN2C(=O)Cn2cnnn2)ccc(O)nc1=O 36315,C1(NC(c2cncc(OC)n2)=O)CN(C(c2cc(C)c(C)o2)=O)C(C)(C)C1 36316,C(=O)(C#CC(C)(C)C)NCCCN(C(=O)CN1CCN(CC)CC1)CC.COC=CC=O 36317,CC1(CNC(=O)CC2CCSCC2)CCCN(C(C2CC3(C2)CC32CC2)=O)C1 36318,c1(C(N(C2CN(C(C3CCC(C)C3)=O)C2)C)=O)ccc(S(=O)(=O)NCC(N)=O)o1 36319,N1(C(CCC=CC)=O)CC(CNC(=O)COc2cc(C)ccc2C)OC(C)(C)C1 36320,Cc1cc2cc(F)ccc2n1CCNC1CC(C)S(=O)(=O)C(C)C1 36321,CC(C)CC(O)CC(=O)N1CC(C)C(C)(CNC(C2(C(C)C)CC2)=O)C1 36322,Cc1ccc(C(=O)NC2CCC(C)N(C(c3ccnc(F)c3F)=O)C2)cc1N 36323,Cc1ccc(CC(=O)NC2CC2CNC(C2C(C)(C)C2(F)F)=O)cn1 36324,C1(CNC(c2c(COC)cccc2)=O)(NC(=O)CSS(C)(=O)=O)CCCCC1C 36325,N1(C(=O)NC(c2cc[nH]c2)C)CC2C(Cc3ccc(Cl)cc3)C2C1 36326,c1(C(N2CCCC(CN(C(C(CC#C)C)=O)C)C2)=O)c(C)nn(CCO)c1C 36327,CC1CCCN(C(=O)CC(C)(C)C#N)C1CCNC(=O)CCc1cc(Cl)no1 36328,C1(NC(CC(C)C2CCCCC2)=O)CCC2(CC1)CC2NC(c1cc(Cl)no1)=O 36329,Cc1cc(C(=O)N(CC(C)C(=O)NCc2nn[nH]c2C2CC2)C)n(C)n1 36330,c1(OC)cc(CC(N2CCC(NC(C3CCCOCC3)=O)C2(C)C)=O)ccc1C 36331,C1(CNC(CCC(=C)Cl)=O)CN(C(c2c(N)cc(Cl)cc2F)=O)CC2(CCC2)O1 36332,CCC1=C(C(=O)NCCN(C2CCCC2)C(C2CCCC(F)C2)=O)SCCO1 36333,Cc1cc(O)ncc1NC(C1CCC(C2CC2)N1C(c1nnn(C)c1N)=O)=O 36334,CC(C)C(CNC(C1CCC(N(C)C)C1)=O)C(=O)N1CCCC(C)C1 36335,C1(CNC(Cc2cccc(OC)c2)=O)CC(F)(F)C12CCC2 36336,N1(C(CCC=C)C(=O)NCCN2CCOCC2)CCN(C)CC2(C)CCCC12 36337,C1(CNC(c2n(C(C)C)ccn2)=O)CC(C)N(C(=O)C(N2C(=O)CCC2=O)C)C1 36338,N1(C(CCC(C)OCC(=O)CN)=O)CC2CCC1C2COCC.c1(OC)nc[nH]n1 36339,Cc1cc(C(N2CC(NC(c3cc(C4CCCC4)[nH]n3)=O)C3CC23)=O)c(C)cn1 36340,c1(C(=O)Nc2c(O)ccc(C)c2)cc2[nH]ccc2cc1-c1ccc(CO)o1 36341,C(=O)(C(CNC(c1oncc1CC)=O)CC(C)C)NC1(CC#C)CCC1 36342,C1(N(C(=O)CC2CCC3CC23)CC)CCN(C(=O)Cc2ccccc2F)CC1 36343,CC1CN(C(c2cc(CCCO)on2)=O)CC(C)C1NC(=O)C1CC1 36344,N1(C(C2CCOC2)=O)CCCC(Cn2cc(C3CC=CCC3)nn2)C1 36345,C=CCC(CC)C(=O)N1CC2CCC2(NC(=O)COc2cncc(Cl)n2)C1 36346,C1(NC(CCCC=C)=O)CC2CC1N(C(=O)CCc1ccsc1Cl)C2 36347,N1(C(C(CC)(C)O)=O)C2CCC1CC(CNC(=O)C(C)(C)Nc1ccccn1)C2 36348,c1(OS(CC2C(C)(C)OCC2)(=O)=O)c(-c2ccccc2)nc2ncccn12 36349,C=Cc1ccccc1N(c1nccn1N)C(c1cscc1C)=O 36350,c1(C(N2CCN(C(c3cn(CC)nc3)=O)C(CO)C2)=O)cccn2c(O)nnc12 36351,CCC(C)(C)C(C)CC(=O)NC1CCC1CNC(=O)Cn1cnc(C#N)n1 36352,CCC(CCC(=O)N1CCC(C(C)(F)F)CC1)OC 36353,C(C(=O)NNC(=O)c1ccc(Cn2cccn2)o1)Oc1cccc(CC#N)c1 36354,C1(C(N(C(CSC)C)C)=O)CC(NC(=O)CC2CCC=CCC2)C1(C)C 36355,C1(CC(=O)NCC(CCOC)NC(=O)CN2CCS(=O)CC2)COC(C)(C)CO1 36356,C(=O)(C(F)CC(C)(C)NC(=O)CCCCCF)N1CCCC(C(C)C)CC1 36357,c1(NC(C2N(C(CSCC(C)=O)=O)CCC2C)=O)cnc(F)cc1C 36358,C1(NC(CC2N(C)CCC2)=O)COCCN(C(=O)CCSCC(N)=O)C1 36359,c1(OC)ccc2[nH]cc(C(=O)NC(C)CC(C)NC(=O)CSC3CC3)c2c1 36360,N1(C(C(C)OCC(C)C)=O)CCC2(CCC2)C(NC(=O)C=C2CC2)C1 36361,C#CC1CN(C(=O)Cc2ccc(Cl)s2)CCN1C(c1cc(C(C)(C)C)[nH]c1C)=O 36362,C#CC1(C(=O)NCCC(=C)CNC(=O)CN2CCC(OC)C2)CCCCC1 36363,Fc1cc(F)c2[nH]c(=NC3CCCOC3)[nH]c(=NCCCn3nccn3)c2c1 36364,C(CCCC(C)(C)C)c1nnc(OC(C)(C)C)o1 36365,c1(CNC(CC2N(C(CC(C)c3ccco3)=O)CC2)=O)ccc(O)cc1 36366,C1(NC(CCOC)=O)CC=C(C(=O)NCC2CC3C=CC2O3)C1 36367,N1(C(Cn2c(C)nc(C)n2)=O)CCC2(CC1)CCN(C(C1(C(F)F)CC1)=O)CC2 36368,N1(C(C(=O)NCCCC)C(C2CCOC2)OCC)CCC2(CC1)NC(=O)NC2=O 36369,c1(C(N(C(CCNC(c2c(CC)ncnc2)=O)C)C)=O)ccc(C(C)C)nc1C 36370,CN1CCN(C(c2cc(CNC(=O)CCc3ccsc3)[nH]n2)=O)CC1CO 36371,Cc1nc(N)c2c(C)c(C(=O)NCc3ccc(CNC(=O)C(N)=O)cc3)sc2n1 36372,N1(C(C(C)SCC)=O)CCc2sc(CNC(c3cc(F)c(C)cc3O)=O)nc2C1 36373,c1(CC)ncc(C(=O)NC2COCC2NC(=O)CCC2CC2(F)F)c(C)n1 36374,C1(C(=O)Nc2scc(C(=O)OCC)n2)C(C2CC2)CCN1C(C1CCCO1)=O 36375,C(C)(C)(C(=O)NC1CCC1C(=O)NCCCN1CCCC1C)SC 36376,C(=O)(CCCCCC(C)C)NCC(CC=C)NC(C12CC(CC(C)O1)C2)=O 36377,N1(C(=O)Nc2cc(C)c([N+](=O)[O-])cn2)CCC(N=c2[nH][nH]c(=N)[nH]2)CC1 36378,c1(C(=O)NC2CCN(C(C3CCNC(=O)C3)=O)CC2)ccnc2ncccc12 36379,C1(CN(C(=O)Cc2cccs2)C)CN(C(c2ccon2)=O)CCO1 36380,N1(C(C(COC)OC)=O)CCC2CCN(C(c3ccc4cncn4c3)=O)CC2C1 36381,c1(CC)nccn1CC(c1ccccc1)NC(=O)NCCC(O)C1CCC1 36382,C#CCN(OC)C(=O)CC1(NC(c2ccn(CC)n2)=O)CCC1 36383,CCC(O)C(C)(C)C(=O)NCC1CCN(C(=O)CSCCC(C)C)C1 36384,Cc1c(C(=O)N(CC(O)CNC(C2COC(=O)N2)=O)C)[nH]c2c(C)cccc12 36385,C1(CC)CN(C(c2c(F)cccc2Cl)=O)CCN1C(c1cc(CN(C)C)c[nH]1)=O 36386,CC1(C)C(NC(C2COC(=O)C2)=O)CCN1C(=O)COC1CCCC1 36387,c1(CNC(C(CCC)CC)=O)ccc2c(c1)CN(C(C1CCN1S(C)(=O)=O)=O)C2 36388,C#Cc1ccc(NC(c2cnn(C3CC3)c2C)c2nnnn2CC)c(C)c1 36389,C1(CCN(C(CNC(CCC)=O)=O)C)CCCCN1C(c1conc1C)=O 36390,N1(C(C(=O)N(C)C)=O)CC2CCCCC2(CNC(C2(C)CCCCNC2=O)=O)C1 36391,c1(NC(C(CC)(C)OC)c2nnnn2CCCF)ccc(C)c(S(C)(=O)=O)c1 36392,O=C1CCC(C(=O)N(C2CC(C(=O)OC)C(O)C2)C(=O)CN2CCCCCC2)=NN1 36393,C(=O)(C(C)(C)CCCNC(c1cccc2c[nH]nc12)=O)NC1CC(C#C)C1 36394,C#Cc1ccc(C(N2CC(C)CC2C(=O)Nc2cnn(C(C)C)c2)=O)cc1C 36395,Cc1nc[nH]c1CC(O)C(=O)N(C)CC1CCN(C(=O)CC2C3CCCC23)C1 36396,C(C)(N=c1[nH]c(=NCC(CO)c2cccnc2)c2c(F)cccc2[nH]1)C1CC(=C)C1 36397,C1(C(=O)NC(CC)CNC(c2snnc2C)=O)CCN(S(=O)(=O)NC)CC1 36398,C(=O)(C1=CC2C=CC1C2)NC1CCN(C(C(C)OC(C)(C)C)=O)C1C(C)(C)C 36399,C1(CNC(c2c(OC)n(C)nc2)=O)C(C2CC2)CCN1C(c1nnn(C)c1C)=O 36400,C1(C(=O)NC2(CNC(Cc3scc(C)n3)=O)CCOC2)CCc2c(cnn2C)C1 36401,n1(CC)ccnc1C=CC(=O)NC1CC(CNC(=O)CN(C2CCSC2)C)C1 36402,C(CCCCNC(c1ccn(C2CCOCC2)n1)=O)N(C(C)C)C(c1cnns1)=O 36403,Cn1cc(C(=O)NC2CCCN(C(=O)CCc3ccncc3)C2)c(O)n1 36404,NS(=O)(=O)c1ccc(C(=O)NC2(CNC(=O)C(F)(F)C3CC3)CC3CCC2C3)o1 36405,N1(C(C(CC)C)=O)CC(CNC(c2sccc2C)=O)OC(C)(C)C1 36406,Cc1cc(N2CCCC(C)(NC(=O)CCC(F)(F)F)C2)ccc1[N+](=O)[O-] 36407,C(=O)(C(O)CCC(F)(F)F)NC1CCCC(NC(c2cn(CC)nc2)=O)CC1 36408,N1(C(C(C)OCC(C)C)=O)CCOC(C(N2CCCC(C)(C)C2)=O)CC1 36409,c1(NC(C)=O)cnc(C)c(C(N2CCCC2CNC(C2OCC2(C)C)=O)=O)c1 36410,C(N=c1[nH]c(=NC2CCCN(C)C2)c2cc(Cl)ccc2[nH]1)C1CC(=C)C1 36411,c1(C(=O)O)cc(F)c(C(C2(CO)CC2)NS(=O)(=O)C(F)(F)F)cc1F 36412,Cc1sccc1C(=O)NCCC1CCCN1Cc1csc(-c2ccco2)n1 36413,CC1CN(C(c2ccc3sccc3c2)=O)CC(C)CN1C(c1cscn1)=O 36414,N1(C(C(C)OCC)=O)CC(NC(=O)CCc2cnc(O)[nH]2)C2(CCOCC2)C1 36415,c1(OCC(=O)NC2CC(C)(NC(C(C(C)C)SCC)=O)C2)cc(C)ccc1F 36416,CCC(C)C(C)CCNCC(=O)NCC(=O)Nc1cccc(C(F)(F)F)c1 36417,c12cc(N(C)C)ccc1OC2=O.C1(N(CC)CC)CCS(=O)(=O)C1 36418,c1(C(C)(C)C)nc(N2CCCCC2CNC(c2cncc(F)c2)=O)cc(Cl)n1 36419,CCC(C)CC(C)C(=O)N(CC(=O)NC1C2CCN(CC2)C1C)C1CCC1 36420,c1(C(C)C(=O)N2CC(C(C)N)C2)c[nH]c2ccccc12 36421,C1(O)(CNC(C(C)(F)F)=O)CCCN(C(C23CCC(CF)(C2)OC3)=O)CC1 36422,c1(C(c2n(CC(=C)C)nnn2)NCCc2cccc(F)c2)cc(F)c(F)cc1F 36423,S(=O)(=O)(C1CCN(C(C2CCS(=O)(=O)C(C)C2)=O)CC1)NC 36424,c1(OC)ccc(CN2CC3CC3(C(=O)Nc3ccc(C4CC4)nc3)C2)c(C)c1 36425,C1(C(C)NC(Cn2cc(C(=O)OC)nn2)=O)CCCN(C(C2(CO)COC2)=O)C1 36426,N1(C(c2coc(CO)c2)=O)CCCN(C(=O)C2=C(Cl)CCC2)C(CO)C1 36427,c1(CC)cc(C(=O)NCCCC(=O)NC(CO)(CO)CO)c(C)o1 36428,Cc1nccc(N2CCCC2)n1.C12(CCCC1)C(=O)NC(C)CN(C(C)C)C2=O 36429,C1(O)(CN(C)C(c2ns[nH]c2=O)=O)CCCN(C(c2ccc(OCF)cc2)=O)C1 36430,N1(C(C(CC)OCC)=O)CCC(O)(CCNC(=O)CCc2nccs2)C1 36431,c1(C(N2CCN(C(CCC=C)=O)C(CC)C2)=O)cc2ccc(OC)cc2nc1C 36432,C1(NC(c2nc(C(C)=O)sc2)=O)CCC(C)(CNC(c2ccc(CO)s2)=O)C1 36433,C1(C(=O)NC(CN(C(c2cncc([N+](=O)[O-])c2)=O)CC)C)CCCCC(C)(C)C1 36434,c1(NC(c2cc(-c3c(OCOC)cc(F)cc3)[nH]n2)=O)c(C)cc(C#N)cc1Cl 36435,c1(OC)ccc(Cl)c(OC)c1C(=O)NCC1(C)CN(C(c2cc(C)nn2C)=O)C1 36436,N1(C(CN(C(c2n[nH]c(O)n2)=O)CC)=O)CCCC1C 36437,c1(C(N(CC(=O)OCC)C2CC2)=O)occc1CNC(c1cocc1C)=O 36438,Cc1cn(C)nc1C(=O)NCC1CCCN1C(c1c(C)ccn1C)=O 36439,C1(CNC(=O)C(N2CC3CCCC(C2)C3(F)F)=O)CCCC12NC(=O)NC2=O 36440,N1(C(C2CCOC2)=O)CCCN(C(=O)Cc2cscn2)C(c2ccccc2)C1 36441,C1(C(=O)NCCCCNC(CSCCC)=O)(N(C)C)CCCCC1 36442,C(CC(O)CC(=O)NC1CC2(C1)CC(NC(=O)CCc1nnc(C)n1C)C2)SC 36443,C1(NC(C(C)N2CCCC2)=O)CC2CCC1(C(N1CCCC1C)=O)C2 36444,c1(C(N2CC3N(C(c4c(OC)nsc4)=O)C(CC3)C2)=O)csc2c(O)ccnc12 36445,C1(c2n(CCCOC)nnn2)(Nc2cc(C)cc(F)c2)CC2CC(OC)CC12 36446,c1(C(N(C2CCN(C(c3cccc(F)c3I)=O)C2)C)=O)cc(F)c(Cl)cc1Cl 36447,C1(CC)(CO)CCN(C(=O)NCCNC(c2ncccc2N(C)C)=O)C1 36448,Cc1cc(C)c(C(N2CCOC(CCNC(=O)C(C)(F)F)C2)=O)c(O)n1 36449,C(CCC(C)CC(=O)NC1CN(C(=O)Cc2cocn2)CC12CC2)=C(C)C 36450,CC1(C)CN(C(C2(c3ccno3)CC2)=O)CCN(C(C2(C)CCC(=O)NC2)=O)C1 36451,c1(CNC2CC(NC(c3cn(CCC)nc3)=O)C2)cc(OCC)ncn1 36452,C#CCCCCC(=O)NCC1CCN(C(=O)CSC)C1 36453,N1(C(C=CSC)=O)CC2CCC(CNC(C3C4CCCCCCC34)=O)(C2)C1 36454,C1(OC)CC(NC(=O)C(C)C(F)(F)F)CN(C(c2c(C)nc(C3CC3)n2O)=O)C1 36455,c1(C(=O)NC2C(NC(C3(CCN(C)C)CC3)=O)CC2)cccnc1C(F)(F)F 36456,c1(NCC2C(C)CN(C(c3ccc(=O)oc3)=O)CC2)c(F)cccc1[N+](=O)[O-] 36457,c1(CC)ccc(C(=O)NC(C2CCCCC2)CNC(C2CSCCS2)=O)s1 36458,N(C(=NCc1cc(C)nn1C)N1CCc2ccc(Cl)cc2C1)C(C=C)C 36459,Cc1cccc(C(=O)NC(C)(C)C)c1NC(=O)C(N1CCCC(CS(N)(=O)=O)C1)C 36460,N1(C(C(COC(C)C)NC(C2OCCCC2(C)C)=O)=O)CC(C)CC(C)(C)C1 36461,Cc1c(C(N2CCCC2CN(C)C(C2(O)CC2)=O)=O)sc2cc(F)ccc12 36462,C12(NC(c3nocc3Cl)=O)CCCC1N(C(c1ccc(OC(F)F)cc1)=O)CC2 36463,C1(CNC(C(C)(C)OCC)=O)CCN(C(c2coc3c2COC3)=O)CC1O 36464,C1(C(=O)NCCC2(NC(COC)=O)CCC2)CCN(c2ccncc2)C1 36465,c1(C(=O)NC(C2CCCN2C(=O)C=C(Cl)Cl)(C)C)cc(P(C)(C)=O)cs1 36466,Cc1cc(F)c(C(=O)NCC(O)CN(C(=O)Cc2c[nH]ccc2=O)C)cc1F 36467,Cc1cccc(-c2csc(C(=O)NC(C)C(N)=O)c2)n1 36468,Cc1[nH]c(C)c(C(N2CCOC(CNC(=O)CC(C)C(F)F)C2)=O)c1C 36469,c1(C(N2CCC(N(C(C3(OC)CCCC3)=O)C)CC2)=O)cc(S(N)(=O)=O)c(C)o1 36470,C1(CC(=O)NCc2c(C)cc(C)s2)CCCN(C(c2ccccc2)=O)CC1 36471,C(=O)(C(C(=O)Oc1cccc(OS(C)(=O)=O)c1)c1ccccc1)OCC 36472,C1(CNC(c2ccc(OCCF)cc2)=O)CN(C(=O)COCCCF)CC12CC2 36473,C#CC1(O)CC(C(=O)NC2CCOC(c3ccncc3)C2)C1 36474,N1(C(c2n(CC)nc(C)c2)=O)CCN(C)CC1CNC(=O)CC(C)c1ccco1 36475,N1(C(COC)=O)CCC(CNC(=O)C(c2cncnc2)C)C(F)(F)C1 36476,c1(C(=O)NC2CC(CCNC(C(CCOC)OC)=O)C2)cnc2[nH]c(O)nc2c1 36477,C(C(C(=O)NCC1CC(C)(NC(=O)C(C)Sc2nncn2C)C1)NC(C)=O)OC 36478,C1(C(=O)NCc2cc(C)ncc2)COC2(C1)CN(C(C1CCC(=O)C1)=O)C2 36479,NC(=O)CCC(C(=O)N=c1ccn(-c2ccncc2)[nH]1)n1cc2nnncc2n1 36480,c1(OCC=C)ccccc1C(=O)NCC=CCNC(C1CCCC1O)=O 36481,C(=O)(N=c1[nH][nH]c2c1CN(C(c1ccc3[nH]c(C)cc3c1)=O)C2)SC(C)=O 36482,C1(C)(C(N(CCNC(C2CC3C(C2)C3(F)F)=O)CC)=O)C2CC3CC(C2)CC1C3 36483,C1(CCNC(C2CCN(CC)C2)=O)CCN(C(=O)CSCC2CCCCO2)CC1 36484,C(=O)(C(C)(C)c1cccs1)NC(C1CC(NC(=O)CCc2ncc[nH]2)C1)C 36485,C1(NC(CC(=O)N(C)C)=O)CN(C(=O)CCCc2ncc(Br)cn2)CC1O 36486,c1(C(=O)NC23C(CN(C(Cc4ccc(C)s4)=O)C2)C3)ccc2ncc(=O)[nH]c2c1 36487,CCCC(C(=O)N1CCC1C(=O)N(CC(C)(O)C1CC1)C)OC 36488,CC1CCN(CC(=O)NCC2CCC(N(C)C(C3(C4CCC4)CC3)=O)CC2)CC1 36489,C(=O)(C(C(C)C)NC(c1ccco1)=O)N(C1CCN(C(CC(C)C)=O)C1)CCO 36490,CC1CN(C(C2CCC(N(C)C)CC2)=O)CC1NC(c1nncs1)=O 36491,N1(C(C(C)c2ccsn2)=O)CCC2(CCC2)C(NC(=O)CCC2CC2)C1 36492,C1(O)(CC)CCOCC1.C1(C(C)C)CCN(C2C(C(=O)O)C23CC3)C1 36493,N1(C(C2(CC)CN(C(C(CCC)NC(C)=O)=O)C2)=O)CCC2(CCCN2C)C1 36494,c1(C(N2CC(OCCNC(CS(CC)=O)=O)C2)=O)cc(C(=O)OC)cc(O)c1 36495,c1(C(=O)NCC(CC)NC(C2CCCNS2(=O)=O)=O)cc(S(C)(=O)=O)c(C)o1 36496,C1(C)(CNC(NCC(CC)(C)C)=NCC2CCCCO2)CCCC1(F)F 36497,N1(CC(=O)NC2CCC(CNC(C3(N(C)C)CCC3)=O)C2)C(=O)CC(C)(C)C1=O 36498,C1(C(=O)NCC(C(=O)N2CC(OC(C)C)C2)O)CC2CCC2C1 36499,c1(C(N2CC(C)C(C(=O)NCC3(CO)CCCCC3)C2)=O)cc2ncccc2[nH]1 36500,C(CC(O)C(F)(F)F)NC(C1CCC(NC(c2cc(C(C)=O)[nH]n2)=O)C1)=O 36501,Cc1nn2c(c1CNC(C1(F)C(C)(C)C1(C)C)=O)CN(C(c1ccccc1)=O)CC2 36502,c1(C(=O)NC2CCC(NC(C(C)n3ccnn3)=O)CC2)nn(C)c2c1CCC2 36503,C1(CNC(C2(SCC)CC2)=O)CCN(C(C2C3CCCCC23)=O)CC1 36504,CC1=C(C(=O)N2CC(O)CC2C(=O)NCCC2CC=CCC2)CC1 36505,c1(C(=O)NCc2c(C(N(C(CCC)C)C)=O)scc2)cc(OC)n(C)n1 36506,C1(CC)COCCN(C(c2cc(CCNC(=O)C(C)SC(C)C)on2)=O)C1 36507,C1(C)(CC(=O)OC)CCN(C(c2ccc(C)c(I)c2)C(=O)NCC(C)C)CC1 36508,c1(C(=O)NCC(CC)(CC)NC(c2ccn(C)n2)=O)c(O)cc(F)cc1F 36509,C(=O)(C(O)Cc1ccccc1)NCCCN(C(=O)CC1CCCO1)C(C)C 36510,c1(C(c2nc[nH]n2)CC)ccc(S(=O)(=O)CC)cc1 36511,C1(NC(CC(C)(C)OC)=O)CN(C(C23CCC(N=[N+]=[N-])C2C3)=O)CC(C)(C)C1 36512,C1(NC(c2c(SCc3nc(C)on3)cccc2)=O)CN(C(N)=O)CCC1C#N 36513,c1(NC(C2CC(F)(F)C2)CO)[nH]c(=NC2CC2c2ccccc2)nc2scnc12 36514,Cc1ccc(C)c(C(=O)NC2CC(C)N(C(C3CC(O)(C(F)(F)F)C3)=O)C2)c1 36515,c1(C(C(C)NCc2cnn(C(C)(C)C)c2)O)ccc(F)cc1F 36516,C=CC(CC)CC(=O)NCCC1CSCCN1C(c1n[nH]c(C2CC2)c1Cl)=O 36517,c1(OC)nc(C(=O)NCC(C)CNC(=O)CCC(=O)c2ccccc2)cc(O)n1 36518,NS(=O)(=O)c1cc(CN2CCC3(C2)CC3(F)F)c(Cl)cc1F.C12(CC1)C(=O)NC2 36519,C(C(C)NC(c1cc(C)n(C)n1)=O)(C(C)C)NC(c1cnc(CCCC)s1)=O 36520,C(=O)(C(CC(F)F)C1CCC1)NC1CC(CNC(=O)CCn2cncn2)CC1O 36521,C1(F)(CNC(C(C)S(N)(=O)=O)=O)CCCN(C(C2NC(=O)OC2(C)C)=O)CC1 36522,c1(C(N2CC(CCNC(=O)C(C)(O)C(C)C)(OC)C2)=O)ccc2nnn(C)c2c1 36523,N1(C(c2c(OC)cccc2)=O)CCC(C)C(CNC(=O)CCc2cccs2)C1 36524,CN1CCC(C(N2CC(O)(CNC(C3CCCC34CCC4)=O)C2)=O)S1(=O)=O 36525,Cc1cc(C)n(C(C)CNC(N2CCCC2Cc2ccncc2)=O)n1 36526,c1(OC)cc(F)c(F)cc1NNC(=O)NC(c1ccc(Br)cc1)C 36527,c1(C(=O)NCC(C2CCC2)NC(CC(=O)NCC)=O)ncncc1Cl 36528,C(CCCCC(=O)NCC1(C(C)(F)F)CC1)N(C(c1ccc(CC)cc1)=O)C 36529,C1(NC(C2CCOC(C)C2)=O)CCCC(C(=O)NC2(OC)CCOC2)C1 36530,c1(CNC(N2CCCC2CCC2CCOC2)=O)cc(Cl)ccc1Br 36531,C(=O)(C(O)C(C)(C)C)N1C(C(=O)NCC2CC3CCC3C2)CC(C)C1 36532,Cn1nnnc1SSCCCNC(CCNC(=O)COC1CCOC1)=O 36533,c1(CC)c(C(N2CCCCC2CN(C(=O)CCc2nncn2C)C)=O)ccn1C 36534,C1(C)(CC(=O)N(CCCNC(C2(CC(F)(F)F)CC2)=O)CC)CCS(=O)(=O)N1 36535,C(CCCCC(=O)N(CC(C)O)CCNC(C1CC(O)CN1C)=O)OCC 36536,C(=O)(C(C(C)C)OC)NCCC1C(NC(C(COC)C)=O)CCC1 36537,C1(NC(C(C)NC(C2CCCC2)=O)=O)CCN(C(=O)CC(C)(C)C2CC2)CC1F 36538,N(C1CCCc2ccoc21)C(C1N(C(=O)Cn2ncccc2=O)CCN(C)C1)=O 36539,C1(CNC(C2(CCC)CC2)=O)CN(C(c2snnc2C2CC2)=O)CCC1(C)C 36540,C(C(C)C(=O)NCC(O)CNC(=O)C(C)OCc1ccccc1)NC(C)=O 36541,N1(C(C)C)CCCN(C(C2CCC(C(C)C)N2C(=O)C2=CCOCC2)=O)CC1 36542,CC1=CCSC1C(=O)NCc1ccsc1C(=O)NCCC(C)N(C)C 36543,C(=O)(CC1=NNC(=O)C1)NCC1N(C(c2c(C)cc[nH]c2=N)=O)CCCC1 36544,C1(O)(C(C)C)CCCN(C(=O)CCS(C)=O)C1.c12cn(nn1)CCC21CC1 36545,c1(N2CCC(N(C)C(=O)NC3CCCC(OC)C3)C2)ccc([N+](=O)[O-])cc1C#N 36546,c1(C(=O)NCC(C2CC2)NC(c2ccc(CC)c(N)c2)=O)cccc2scnc12 36547,c1(C(=O)NCCNC(C2CC(C(F)(F)F)CO2)=O)cc2ncccc2s1 36548,C1(CNC(Cc2c(C)noc2)=O)CN(C)CCN1C(c1cccc(=S)n1O)=O 36549,c1(C(N(C)CC2CCN(C(C3C(C=C)CC3)=O)C2)=O)cc(Br)c(OC)cc1N 36550,c1(CC)cccc2[nH]c(C(N3CC(CNC(C4COCCO4)=O)C(O)C3)=O)cc12 36551,CC1=CCC(C(N2CC(O)(C(C)(C)CNC(=O)CC(C)(C)C)C2)=O)CC1 36552,c1(C(N2C3(C(N(C4CCCCC4)CCC)=O)CC(C2)C3)=O)cc2ccccn2n1 36553,C1(NC(C(C2CCC2)OCC)=O)CC(OC)CN(C(c2cccc(CC)n2)=O)C1 36554,c1(C(CC)C)nccc(N2CC(C)(C)C2C2CCN(C(c3cncs3)=O)CC2)n1 36555,C1(C(N(CCNC(CC2(C(=C)F)CCC2)=O)C2CC2)=O)CCN2CCOCC12 36556,c1(C(=O)Nc2cccc(CNC(CCN(C)CCO)=O)c2)coc2ccccc12 36557,N1(C(C2CCC(CC)C2)=O)CCC(C=CC(=O)NC(CCO)C(F)F)CC1 36558,N1(C(C2CC(C#C)(O)C2)=O)CC(NC(c2cnn(CC(F)(F)F)c2)=O)CC1(C)C 36559,C(=O)(C(CC)CC=CC)N1CC(CN(C(CC2CC(=C)C2)=O)C)OCC1 36560,N1(C(c2ccc(CC)s2)C(=O)NCCCC2CC2)CC2C(=O)N(C)C(=O)C2C1 36561,C1(C(N(c2ccsc2)CC)=O)CN(C(C2CCC3(CCC3)O2)=O)C2(CCC2)C1 36562,C1(C(=O)NC2CCC(C)(CNC(c3cnc(C)nc3)=O)C2)CCC(C)(C)CC1 36563,C(=O)(CCCCCCCCC)NCC(CNC(C1C(=C)CC1)=O)(C)C 36564,c1(C(N2CCC3(CCN(C(C45CC(F)(C4)C5)=O)C3)C2)=O)cnc2ncnn2c1O 36565,CCC(C)CC(C(=O)NC(C)C(C)SC)NC(c1cnc2n1CCC2)=O 36566,CCC(CC)C(C)C(=O)NC(C)(C(=O)NCC1=CCCCC1)C1CCC1 36567,C1(O)(C(CNC(C2(CC)COC2)=O)(C)C)CN(C(=O)C(c2cnccn2)C)C1 36568,C1(CNC(c2c(C)scc2)=O)C(C2CC2)CCN1C(c1coc(C(C)C)n1)=O 36569,C1(NC(c2c(C#C)c[nH]n2)=O)CC2CC1CN(C(=O)CC1CCS(=O)(=O)CC1)C2 36570,C(=O)(C(C)C(C)(C)O)NCC(C)NC(c1ccc(OCC(F)F)cc1)=O 36571,CC1CCC(NC(=O)C(C)(C)c2cncnc2)CN1C(=O)C=Cc1ncc[nH]1 36572,C(CC#N)(C(=O)C(C)OC(=O)NC(C(=O)OC)C)NC(=O)OC(C)(C)C 36573,C1(C(N(CCOCCO)CC)=O)CC2(CC2)CN1C(=O)C(C1CCCCO1)C 36574,N1(C(CSCCC)=O)CCCC2C1CCCN2C(=O)CCC(=O)OC 36575,CCC(C)(C)CC(=O)N(CCCNC(C1CSCN1C(=O)C(C)CC)=O)C 36576,C1(O)(C(=O)NC2(CNC(=O)Cc3cc(C)ns3)CC(OC)C2)CC2CCC1C2 36577,C#CCC(CC#C)NC(=O)C(CNC(=O)C=CC1CCOC1)N(C)C 36578,N1(C(C(N(C)C(c2cc(O)cc(=O)o2)=O)C2CC2)=O)CCC(F)(F)C(CO)C1 36579,C12CC(C1(C)C)NC2.c1(C(=O)NC2C(C(=O)OCC)CC2)ncoc1C1CC1 36580,C1(CC)(NC(=O)CC(c2ccc(SC)cc2)C)CCN(C(=O)C(C)(C)CO)CC1 36581,CC(CC(F)F)C(=O)N(C1CCC(NC(=O)C(C)N2CCC2)CC1)C 36582,N1(C(CCCCC)=O)CC2CCC(C1)C2NC(=O)COC1CCCC1 36583,C1(CCOC)CCCCN1C(N1CCC(C)(O)C1)=O 36584,C1(N(C=O)Cc2nscc2Br)CCc2nncn2C1 36585,c1(-c2cccc(C)c2)nnc2n1CC(C(=O)NCC(C)(C)C(C)(F)F)CC2 36586,CC1(C)OC(=O)CC1C(=O)NC1CCCN(C(=O)CSCC(F)F)C1 36587,N1(C(C(CCNC(C2(CC#C)CC2)=O)O)=O)CC2(C1)CC(C)(F)C2 36588,N1(C(c2c(C)coc2)=O)CCC2(CC1)CN(C(C1(C)C=CCCC1)=O)CC(C)O2 36589,C1(O)(C(=O)NC2(CO)CN(C(CC3CC(=C)C3)=O)C2)CCN(C(=O)OC(C)(C)C)C1 36590,CCCC(C(=O)N1CC(CNC(c2cocn2)=O)(COC)C1)C(C)C 36591,C1(NC(=O)CCC2CCCCC2)CC(F)CN(C(=O)C(Cl)(Cl)Cl)C1 36592,C1(NC(c2c(C(C)C)nns2)=O)CCN(CCNC(C2CC2(Cl)Cl)=O)CC1 36593,N(C(=NCCC(=O)NC1CCCCC1C1CC1)NCc1ccccc1C#N)CC 36594,C(CCN=c1cc(C)nc(CC)[nH]1)N(CC)CC.c1ccc(C(F)(F)F)cn1 36595,C1(NC(c2cscc2C2CC2)=O)CC2CCC(C1)N2C(c1ccns1)=O 36596,N1(C(C(=O)NCC)=O)CCC2(CC1)COC(CNC(c1c(Cl)nn(C)c1C)=O)C2 36597,Cc1c(Cl)ccc(C(=O)N(C2CCCN(C(c3cccc(=O)n3C)=O)C2)C)c1O 36598,C1(NC(COC2C(CC)CCCC2)=O)CCN(C(c2cc(O)cs2)=O)C(C)C1 36599,Cc1nc(NCC2(O)CCCN(C(c3cnn4ncccc34)=O)C2)c(C)c(O)n1 36600,C(=O)(C(C)(c1ccccc1)OC)N(C1(CC(=O)NCC2(C(=O)OC)CC2)CC1)C 36601,Cc1nnccc1C(=O)NOCc1cccnc1N1CCN(C)CC1 36602,c1(C(=O)OC)nnc(C(C)NC(=O)OCc2nnc(C)o2)s1 36603,n1(CC(=O)NCC(C2CC2)NC(c2ccccc2)=O)nc(Cl)ccc1=O 36604,CC1CN(C(c2sccc2-n2cnnn2)=O)CCN1C(C1CC2(CCOC2)C1)=O 36605,c1(CN2C(C3CCN(C(C(CC=C)C)=O)CC3)CCC2)ccc([N+](=O)[O-])cc1F 36606,c1(C(N2CCC(C)(c3cn[nH]c3)CC2)C(=O)NC(C)(C)C)cc(S(N)(=O)=O)cs1 36607,Cc1ccc2c(C(=O)NC3CCC(C)N(C(=O)CCOC4CC4)C3)ccnc2c1 36608,c1(C(C)CNC(=O)Nc2ccnn2CC2CC2)ccc(Br)cc1F 36609,CC1CCC(NC(=O)CC2(N3CCCC3)CC2)CN1C(c1cc(N)ccc1F)=O 36610,C1(CN(C)C(C2(C(N)=O)CCC2)=O)CCN(C(c2c[nH]nc2C2CCOC2)=O)C1 36611,C1(C(N(C2CCN(C(c3conc3C3(C)COC3)=O)C2)C)=O)COC(=O)N1 36612,c1(C(=O)NCC(CCCC)NC(=O)C(C)SCC)ccnc(F)c1OC 36613,c1(CC)cc(C(N2CCC(CCNC(=O)CC3CCCO3)C2)=O)ccc1OC 36614,N#Cc1c(C(=O)NC2CC(NC(c3n[nH]c4c3COCC4)=O)C2)cccc1F 36615,N1(C(C=C(C)C)=O)CCCC(C)C1C(=O)C(C)N(C)C 36616,C1(C(=O)Nc2ncoc2-c2ccon2)CN(C(=O)CCN(CC(F)F)CC)CC1O 36617,c1(OC)ccccc1C(=O)NCC1CC(NC(=O)C(c2ccccn2)O)C1 36618,c1(CC(=O)NCC2(CNC(C3C(C#N)C3)=O)CC23CCC3)cccc2cnccc12 36619,Cc1cc(C(=O)NCc2cc[nH]c2C(=O)NCCc2cnn(C)c2)cc(C#N)c1 36620,N1(CC)CCCC(C(=O)NC(C)CN(C(c2conc2C2CCC2)=O)CC)C1 36621,N1(C(C=CCCC)=O)CCCC(C)C1CCNC(=O)Cn1nc(C)n(C)c1=O 36622,C1(OC)CC2(C1)CN(C(=O)C(O)CCNC(=O)Cc1cncs1)C2 36623,C(CN=C(NCc1cc(O)cc(O)c1)NCc1cc(C)ccn1)N(CC)CC 36624,c1(CC(=O)N(C2CC(C(=O)NCC(C)Cc3cn[nH]c3)C2)C)cccn1C 36625,c1(C(=O)NCCCOCCN(C(=O)CC2COC(=O)C2)C)c(Cl)cnn1C 36626,c1(C(=O)NC2CC(N(C(=O)CCc3ccoc3)C)C2)cc(Br)c(F)cc1N(C)C 36627,C1(OC)CC(NC(C2CCC(=O)N2C)=O)CN(C(c2c(SC)cnn2C)=O)C1 36628,C1(C(=O)NC2CCC(NC(c3ccncc3O)=O)C2)CCCC1(F)F 36629,Cc1nn(C2CC2)cc1C(=O)NCC(C1CC1)NC(=O)CNc1ccccn1 36630,C1(C(=O)NCC(C)NC(CC2C(OCC)COCC2)=O)CC(=O)NC1(C)C 36631,N1(C(CNC(CCC)=O)=O)CC2CCN(C(c3ccoc3Br)=O)CC12 36632,c1(C(N2C(C(=O)Nc3c(OC)cc(C)cc3)CC2)=O)cc([N+](=O)[O-])cc(O)c1O 36633,N1(C(Cc2nc(C)sc2)=O)CCCN(C(=O)Cc2cccc3nonc23)C(C)C1 36634,C(CCC(N)=O)(C(=O)NCC1CCN1C(=O)C=CCN1CCCCC1)NC(C)=O 36635,C(C(COC)C(C)C)NC(c1cccc(C)c1)c1n(CCSC)nnn1 36636,C(=O)(CCC(=O)NN(C)C)NC1CC(C)CN(C(c2cc(O)nc(O)c2)=O)C1 36637,c1(CC)nc(C)c(C(N2CC(C(=O)NC(C)(CO)C3CC3)(CC)C2)=O)o1 36638,C1(C(=O)CC2CC2C(=O)OC)CCCN(C(=O)C(=O)C2CC2)C1C 36639,CC1(C)CCCC(CC(=O)NCC2COCCN(C(c3ccoc3Cl)=O)C2)C1 36640,c1(C(=O)NCC2C(N(C(=O)CCOC3CC3)C)COC2)c(F)cccc1[N+](=O)[O-] 36641,N1(C(C(C)=C2CCC2)=O)CCN(C(c2c(C3CCC3)cnn2C)=O)CC1C 36642,c1(CNC(N2CCC(c3c(C(=O)OC)c[nH]n3)C2)=O)cc(C)n(C)c(=O)c1 36643,C(=O)(C(C)(O)CC(C)C)N1CCC(CCOC)(NC(=O)CCS(=O)(=O)N(C)C)C1 36644,C(=O)(C#CC1CCOCC1)NC1CCC(CC(=O)NCC(C)O)CC1 36645,C(CC(C)C)(C(=O)NCC(C)CN(C(=O)CC1CCC(C)(C)CO1)C)NC(C)=O 36646,C1(C(=O)NC(C2CCCCC2)C#C)COCCN1C(c1ccnc(C)n1)=O 36647,CCCS(=O)(=O)c1ccccc1C(=O)NCCCCCNC(C1CC1F)=O 36648,Cc1nc(C(=O)NC2CC2CNC(=O)C=CC2CCCCCC2)c(C)n1C 36649,n1(COC)nccc1C(=O)NC1CCC1CNC(C1CCC(C(=O)OC)C1)=O 36650,C1(CCNC(c2n(CCSC)nnn2)c2ccncc2)CC2CCC1CC2 36651,c1(OCC)ccc(C)cc1CNC(=NC)NCC1(C#N)CCCC1 36652,Cc1ccc(S(=O)(=O)N2CCC2C(=O)Nc2cc(C)cnc2Br)c(F)c1 36653,N1(c2nnc(CCC)s2)CC2(C)CN(C(=O)CCCCSC)CC2(C)C1 36654,C1(CC(=O)NCCC(C)(C)NC(CC(C)SC)=O)CCOC(C)(C)C1 36655,C1(C2CCN(C(c3cnsn3)=O)C2)CCCCN1C(=O)Cc1ccc(O)nc1 36656,C1(C#CC(=O)NCC2CC2CNC(=O)C=C(C)C(C)(C)C)(CC)COC1 36657,C12(CNC(C3OCCN(C)C3)=O)CCC(CNC(C3CC3[N+](=O)[O-])=O)(CC1)CO2 36658,c1(CN(C(C(C)O)(C)C2CCOCC2)C=O)ccc(Br)cc1OC1CC1 36659,N1(C(C)=O)CCC(CC(=O)O)C(NC(=O)Cc2cc(C)nn2C)C1 36660,C(=O)(NNC(=O)C1OCCC1Cn1cc(C)cn1)OCC 36661,N1(C(Cn2c(C)nnn2)=O)CC(CNC(c2cnn(C)c2Br)=O)CC12CCC2 36662,CC(C)C(O)C(C)C(=O)NCCCC(=O)N1CCC(Cc2ccccc2)C1 36663,c1(CC)ccc(C)c(C(=O)NC(C)C(C)(C)NC(=O)CN2CCSCC2)c1 36664,CC1CCc2nc(C(=O)NCC3CCCC3NC(=O)CC(C)(C)O)ccc2C1 36665,C1(NC(c2nc(-c3c(C)cccc3)sc2)=O)(CNC(=O)C(N)=O)CC2CCC1C2 36666,Cc1ccc(F)cc1CC(=O)NC(C)C(C)(C)NC(C1CC2(CCC2)CO1)=O 36667,n1(CC)nccc1C1OCCC1NC(=O)NCCc1ccccn1 36668,c1(C(=O)NCCCCNC(C2CC(S(C)(=O)=O)C2)=O)cccc2ncsc12 36669,C(=O)(N=c1[nH]nc(C2CC2)s1)N(c1ccccc1CCOC(C)(C)C)C 36670,C1(COC)(NC(=O)C=CC(F)(F)F)CCN(C(=O)Cn2cnc(=N)[nH]2)CC1 36671,Cc1nc(F)ccc1CNC(C1CCN(C(=O)CCC2CC2C)C1(C)C)=O 36672,CCC(N=c1ccnc(NC2CCN(CCC(C)(C)C)CC2)[nH]1)C(C)C 36673,N1(C(CC=CC)=O)CC(NC(=O)C=Cc2ccoc2)CC(F)(F)C1 36674,CC(C(=O)N1CCCC1CCNC(c1c[nH]cc1C(C)(C)C)=O)C(F)(F)C(F)F 36675,CCCCCCCCC(C)C(=O)NC(C1CCN(C(C2(C)CCC(=O)C2)=O)C1)C 36676,N1(C(C(C)NC(CC)=O)=O)CC(=O)NCC1C(=O)NCC1(O)CCN(C)C1 36677,N1(C(COC)=O)CCCC(C)(C)C1CNC(C1(Cc2ccc(F)cc2)CC1)=O 36678,c1(CC(=O)NC2C(NC(c3cc(CCC)nn3C)=O)C2)cn2ccccc2n1 36679,C1(CN(C(C23CC(C(=O)OC)(C2)C3)=O)C)CCCC(NC(=O)CC(F)(F)F)C1 36680,c1(N2CC(C(C)NC(c3cc(C)no3)=O)OCC2)ncnc2scc(C)c12 36681,c1(N2CCC(O)(C(C)NC(c3c(C(C)C)nns3)=O)C2)ncc([N+](=O)[O-])cc1F 36682,C1(C(=O)NC(CCCNC(CCC(=O)NCC)=O)C)COCC(C)(C)O1 36683,N1(C(CCC2CCC(C)O2)=O)CCC(CNC(=O)C(C)C2CC2)CC1 36684,CC(C)C(C)CC(=O)NCC1CC(C(=O)NCC2CC3(CC3)C(=O)O2)=NO1 36685,C1(C(=O)NCC(C)N(C)C(c2cnn(C3CCCC3)c2)=O)OCC1(C)C 36686,C1(NC(c2ccc(OC)c(I)n2)=O)CCc2ncc(Br)n2C1 36687,c1(C(=O)NCCC2CN(C(c3c(CC)nccn3)=O)C2)cc2c(=O)[nH]ccn2c1 36688,n1(CC)cnc(C(=O)NC(CO)C(C)NC(=O)CCNC(C2CCOCC2)=O)c1 36689,C(=O)(C(F)CCC(C)(C)C)NCC1CCCN(C(C(CC)NC(C)=O)=O)C1 36690,Cc1cc(C(N2CCC(F)(CNC(C3CCCN3C3CC3)=O)C2)=O)nnc1C 36691,CN=c1[nH]cc(C(=O)N(C)CCN(C(=O)Cc2cnn(C(C)C)c2)C(C)C)s1 36692,C(c1ccc(F)c(Cl)c1)=CC(N1C(CNC(COCC(C)C)=O)CC1)=O 36693,C1(N(CCCC)C(=O)C=Cc2cscn2)CCN(C(c2cc(C)cs2)=O)CC1 36694,c1(OCC(=O)NCc2ccc(-n3cncn3)cc2)ccc(Cl)cc1[N+](=O)[O-] 36695,C1(C(N(CC(C)(C)N(C)C)C)=O)CCN(C(C2CC(C)(C)C2)=O)CC1 36696,N1(CC(CN(CC(C)C)C(c2ccc(CO)o2)=O)O)C2CCC1CN(S(C)(=O)=O)C2 36697,C1(C2CCOCC2)(NC(C(C(CNC(CC(=O)OC)=O)C)F)=O)CC1 36698,Cc1cc(C)c(C(=O)NC(CNC(C2(O)CCC(C)(C)CC2)=O)C2CC2)c(=O)o1 36699,C(=O)(C1=CC2(CN(C(=O)CCn3cnc(=N)[nH]3)C2)OC1)N(CCCC#C)C 36700,C1(NC(C(CCC)=CCC)=O)CCCC(C(=O)NCCN2CCCOCC2)CC1 36701,C(C(F)(F)C(=O)NC(C)CCC(=O)NCC1CC(OC)C1(C)C)OC 36702,C1(CC(=O)NCCC(CC)CO)CCN(C(C2OC3CCC2C3)=O)C1(C)C 36703,c1(CNC(=O)NCC(c2cccc(I)c2)C)ccc2cnccc2c1 36704,c1(C(C)C)cccc(OC(C)C(=O)NCCCCC(C)NC(=O)C=CCO)c1 36705,c1(C(=O)NC(C(N)CO)C(=O)O)cc(Cl)ccc1I 36706,CCCC(C(=O)NCC1CCCCN(C(=O)CCN2CCOCC2)C1)S(N)(=O)=O 36707,Cc1noc(C(F)F)c1C(=O)NCCN(C(=O)Cc1sccc1Cl)CC(C)O 36708,N1(C(C2(NC(C)=O)CCCC2)=O)CCC(CO)(CNC(C2CC(C)(C)CO2)=O)C1 36709,c1(CC(N2CC(O)(C(C)NC(C3CC(CCC)C3)=O)C2)=O)sc(C)nc1C 36710,c1(NC(c2n(CCC)nnn2)C2CC2(Br)Br)ccc(Cl)c(C(N)=O)c1 36711,c1(C(N2CC(C(C)NC(C=CC)=O)OCC2)=O)c(C)ccc(OCC)c1N 36712,c1(N(C)CC2CCCC2O)nc2c(c(=NCC3CCC=CCCC3)[nH]1)COC2 36713,CCC(C)C(=O)NCC(=O)NCCNC(C1CC(OCCOC(C)=O)C1)=O 36714,N1(C(c2c(C)snc2)=O)C2CCC1C(CNC(=O)CCc1nc(C3CC3)no1)C2 36715,CC1(NC(=O)C=Cc2cccs2)CCN(C(=O)CC(C)(O)C2CC2)C1 36716,C1(C(=O)NCC23CC(NC(c4ccc(CC)s4)=O)(C2)C3)CC(C)(C)C1C(F)(F)F 36717,N1(C(CC(COC)C)=O)CCC2CCCC12C(N1CCCCC(N(C)C)C1)=O 36718,C=C(Br)CC(C)(C)C(=O)N1CC(CNC(=O)C(C)NS(C)(=O)=O)C(C)C1 36719,c1(N2CCC(C)OCC2)ccc(S(=O)(=O)NC2CCCC(C(F)(F)F)C2)c(Br)c1 36720,C(CC(CNC(=O)CN(c1cccs1)C=O)NC(=O)CC#N)OC.c1(O)ccccc1.N 36721,N1(CC(=O)N(CC(C2CCC2)OC)C)C(=O)NC(C)(c2ccc(Br)cc2)C1=O 36722,c1(-c2c(C(=O)NC(C)C(C)n3ccnc3)c[nH]n2)ccc2c(c1)CCCO2 36723,c1(C(N2CCC(NC(CCc3c(C)nccc3)=O)C2)=O)ccc(C(F)F)c(Cl)c1 36724,c1(CC(=O)N(C2CCCC2)CCNC(=O)CCc2ccon2)ccc(Cl)cc1 36725,c1(C(=O)NCCOC)ccc(N)c(OC)c1.C1(=O)CN(CC)CCN1 36726,C1(NC(C2C(CC)N(C(=O)CCC(C)(C)N(C)C)CC2)=O)CC(C)(C)OC1(C)C 36727,C(=O)(C(C)(C)c1ccno1)N1CC(N(CC#C)C(C2CN(C(C)=O)C2)=O)C1 36728,C1(C(=O)NCCOCCN(C)C)CNC(=O)CN1C(=O)CCn1cccc1 36729,C1(C(N(C(C)C)CCNC(C2(CC3CCCC3)CCCC2)=O)=O)CC2C=CC1C2 36730,c1(C(=O)NC2CCC(C)(CNC(=O)C3=C(Cl)CC3)C2)cccn2cncc12 36731,Cc1ccc([N+](=O)[O-])cc1C(N1CCC2CN(C(C3(C#N)CC=CC3)=O)CC12)=O 36732,c1(C(=O)NCCCC2(CNC(C(C)O)=O)CCCC2)nccc2cc[nH]c12 36733,CCCCC(F)F.C(=O)(C(CCS)NC(=O)OCC)OC(C)(C)C 36734,C12(C(N3CCCN(C(=O)COc4ccc(Cl)nc4)CC3)=O)CCCCC1C2(F)F 36735,C1(CC(N2C3CN(C(C4(C=C)CCC4)=O)C(C3)C2)=O)CCc2ccccc2C1=O 36736,C=CC1(C(=O)NCC2(NC(C3CC34CCOC4)=O)CCCCCC2)CCOCC1 36737,Cc1cc(F)cc(C(N2CC(N(C)C(C3CCOCC3)=O)C3(CC3)C2)=O)c1O 36738,C=CCC(Cc1ccccc1)C(=O)NCCCOc1c(F)cccc1F 36739,N1(C(C(C)SCC)=O)CCC(CNC(c2cnccn2)C2CCCC2)C12CCC2 36740,N1(C(C=Cc2cc(C)no2)=O)CC2CCC(N(C(=O)C3=CCCSC3)C)C2C1 36741,c1(C(N2C(C)(C(NOCC=C(C)C)=O)CC(O)C2)=O)nccc2[nH]ccc12 36742,C(CNC(=O)Cc1ccccc1)(C(C)(C)C)NC(CCN(C)CCO)=O 36743,C1(C(=O)NCCCN2CC=CC2)CCC(O)CN1C(c1cc(C(F)F)[nH]n1)=O 36744,N(C(=NCc1ccccc1[N+](=O)[O-])N1CCC(C)(F)C1)Cc1cc(C)on1 36745,c1(Cc2c(CNC(C3SCCCS3)=O)con2)ccnc(C2CCC2)n1 36746,C1(OC)(CNC(c2n[nH]c(C)c2O)=O)CCN(C(c2cncc(C(N)=O)c2)=O)C1 36747,CC1CC2(CCN(C(=O)Cc3cncs3)CC2)CN1C(C1CC12CCCC2)=O 36748,c12cccnc1OC2=O.N(S(=O)(=O)Oc1ccccc1)CC(=O)OC(C)(C)C 36749,N1(C(c2c(C)ccc(C)c2O)=O)CCC2(CC1)CC(NC(=O)CCCF)CO2 36750,c1(C(=O)NCCCN(C(=O)C(C)(C)OCC(F)F)CC)cc(C(N)=O)[nH]n1 36751,N1(C(CC2(OCC)CC2)=O)CCC(CN(C)C(c2cnc(C3CCC3)o2)=O)C1 36752,C1(NC(=O)Cc2ccc(Br)cn2)CC2CC1CN2S(=O)(=O)CCBr 36753,C#CCCCCCC(=O)N(CC(C)C(=O)N1CCC2CC12)C 36754,C(=O)(CC(CC(C)C)NC(=O)CCc1cccn1C)Nc1cc(C)c(O)cc1 36755,C(=O)(C(C)(C)CCCF)NCC(C(=O)NCc1c(C)cc(O)cc1)CC1CC1 36756,N1(C(CCOCC(C)(C)C)=O)CCCC(F)(C(=O)NCC23CCCC2CCC3)C1 36757,C1(CNC(C2CC3(C2)CC3F)=O)COCCN1C(=O)Cn1cnnc1O 36758,CC1CN(C(c2cncc(F)c2)C(=O)NC2(C)CC2)C12CCOCC2 36759,c1(C(=O)NC(CNC(C(c2c(C)nn(C)c2)O)=O)CO)cc(Cl)cc(Cl)c1 36760,CC(=O)C(C)(C)CC(=O)N(C1CCN(C(c2ccccc2[N+](=O)[O-])=O)C1)C 36761,C(CC(=O)NC(C)C(=O)C1CCCC1)(C(C)C)NC(c1ccc(OC)s1)=O 36762,N1(S(C)(=O)=O)CCC(NC(=O)C(Cc2ccc[nH]2)C(N2CC(F)(C3CC3)C2)=O)C1 36763,c1(C(=O)NC2C(NC(=O)Cc3ccon3)CS(=O)(=O)C2)cc2cccc(Cl)c2[nH]1 36764,C1(CNC(=O)CCc2ccc(Cl)s2)CN(C(=O)C(F)=CCCF)CC12CCC2 36765,C(=O)(CCCCCNC(C)=O)NCC1CC(NC(COCCC)=O)C1 36766,C(=O)(C(C)C(C)(C)C)NCCCN(C(=O)C=Cc1cccc(CO)c1)CC 36767,c1(SCC(=O)OC)ccncc1NC(c1cc(SC2CCCC2)on1)C 36768,c1(CN2CC(F)CC(C(=O)NC(CCC)C(=O)NC)C2)ccc(F)c(NC)c1F 36769,C1(CNC(c2c(C)cncc2C)=O)COC(C)(C)CN1C(c1cc(Cl)cn1C)=O 36770,N1(C(C(C)OCC#C)=O)CC2CC1CN(C(c1cc(C3CCCCC3)[nH]n1)=O)C2 36771,C1(NC(C(=Cc2ccccn2)C)=O)C2CCC1N(C(c1cc(C(F)F)no1)=O)C2 36772,C1(C2CC2)(C(=O)NCC(c2ccccc2)CNC(C)=O)CC1 36773,CCCC(C)CC(=O)NCCCC(O)C(=O)NCc1cnccc1Cl 36774,C(CCCC(=O)NCC1C2CCCC12)N(C)C(C1CCCN1C=O)=O 36775,c1(C(N(C)C(C2CCCN2C(C2CC23CC3)=O)C2CCC2)=O)cccc(F)c1 36776,Cc1c(NCCCN2CCCN(C)CC2)nc[nH]c1=NCC1CC2(C1)CC(O)C2 36777,N1(C(C=CC)=O)CCC(CNC(=O)CC2CCNC2=O)C1C(C)(C)C 36778,c1(C(=O)OC)ccc(C(N2CCCN(C(C3CC3(C)C(F)F)=O)CC2)=O)c(C)c1 36779,C1(C)(COC(C(C(C)C)n2cncn2)=O)CCCN(C(=O)OC(C)(C)C)C1 36780,c1(NCCCCC(N)=O)[nH]c(=NCCCC2CC2(Cl)Cl)nc2scnc12 36781,c1(C(=O)NCCCN(C(C=CCCC)=O)C(C)C)c(OC)nsc1OC 36782,C#CCCCC(C)C(=O)N1CCOC(CC(=O)NC(c2n[nH]c(C)n2)C)C1 36783,C1(C(=O)Nc2cc(OC)c(O)cc2)CC12CCN(C(c1cc(O)n(C)n1)=O)CC2 36784,CCS(=O)(=O)c1cc(F)ccc1NC(=O)C(N1CCC2CSCC2C1)=O 36785,Cc1ccc(CC(N2CCC2CNC(=O)CN(S(C)(=O)=O)C)=O)c(Cl)c1 36786,C1(O)(N(C(=O)COC(C)(C)CC)CC#C)CCN(C(c2ccc(NC)cc2)=O)C1 36787,C(=O)(C=C1SCC(=O)N1C)NC1CCN(C(C(C(C)C)C)=O)CC1O 36788,CC1CC(C(=O)NC2(CCNC(=O)Cc3ccc(Br)nc3)CCCC2)=NO1 36789,C(=O)(C1CCc2ccccc21)NCCC(C)NC(C(CC)C(C)(C)CC)=O 36790,c1(CC(=O)NCCC(C)NC(C2CC23CC3)=O)c[nH]c2ccc(Cl)cc12 36791,N1(C(=O)CC2CCCN(C(c3cnn(C(F)F)c3)=O)C2)CCC(CO)C(F)C1 36792,CC(CCCCNC(C1CCCCC1O)=O)NC(c1cnn(CC2CCC2)c1)=O 36793,c1(CC(=O)NCC2C(NC(=O)Cc3sccc3Cl)CC2)ccccc1Cl 36794,c1(CNC(c2cc(C)ns2)=O)nc(C)c(C(=O)N(CC(=O)NC(C)(C)C)C)o1 36795,CC1=NOC(C)(C(=O)NC(CO)C(C)NC(=O)Cn2nc(C)cc2C(F)F)C1 36796,C(C1=NOC2CN(C(=O)C=CS(F)(F)(F)(F)F)CC12)NC(=O)C1=C(Cl)CCC1 36797,C(CCC(C)NC(c1nnsc1C)=O)NC(C(C)OCC)=O 36798,C(c1c(C)noc1C)=CC(N1CCC(N(CCC)C(C2CCCN2C=O)=O)C1)=O 36799,N1(C(C(C)S(N)(=O)=O)=O)CCN(C(C2CCc3nncn3C2)=O)CC(O)C1 36800,N1(C(C(C(C)O)NC(=O)OC(C)(C)C)=O)CCCN(C(c2cncs2)=O)CC1C 36801,Cc1cc(C(N2CC(F)CC2CNC(=O)C2=NOC(C)C2)=O)cc(C(F)F)c1 36802,N1(C(C2(SC)CN(C(=O)C(C3CCOCC3)O)C2)=O)CC(C#N)(CCF)C1 36803,CC(CN=[N+]=[N-])NC(C1COCC1NC(=O)CC1CCOC1)=O 36804,C12(C(N(C)OC3CCCC3)=O)CC(C)(CN1C(c1cc(C(N)=O)co1)=O)C2 36805,Cc1ccc(CNC(c2nnnn2CC(F)F)(C)CC2C=CCC2)c(F)c1 36806,c1(OC)ccc(C(=O)NCC(C2CC3(CCCO3)C2)=O)c(N)c1F 36807,C1(CNC(COc2cc(C)on2)=O)CN(C)CCN1C(c1ccncc1Br)=O 36808,C1(CC)CN(C(c2cc[nH]n2)=O)CCC1NC(=O)Cc1ccccc1Cl 36809,CC(C)(CCCO)C(=O)NC1CCCCC1CNC(c1c[nH]nc1[N+](=O)[O-])=O 36810,C(=O)(C(CNC(C1(C)CC(F)(F)C1)=O)CC=C)N(CC#C)CCOC 36811,Cc1nc(N2CC3C(CNC(=O)CC(C)CC(C)(C)C)C3C2)c2cc[nH]c2n1 36812,c1(CC)ccc(F)cc1C(=O)NC1CC(CNC(c2nn(C)c(C)c2N)=O)C1 36813,N1(C(C(CC)OCC)=O)CC(NC(=O)C(c2cnn(C)c2)C)CC12CCOCC2 36814,C1(C(N2CC(O)(CCNC(=O)COCC(F)(F)F)C2)=O)CCC(C2CCC2)CC1 36815,N1(C(C(=O)OC)=O)CCC(C(F)CNC(=O)Cc2ccc(C(F)(F)F)cc2)CC1 36816,C(=O)(CC(C)c1ccco1)N(CCCN(C(=O)CC#N)C)C 36817,C=C(CNC(=O)COCCNC(c1[nH]ccc1CC)=O)c1ccccc1 36818,C1(NC(C(c2ccccc2)C)=O)CCCCN(Cc2ccncc2Cl)C1 36819,Nc1ccnc2c(C(=O)NCC(C3CCCCC3)NC(C3CCCSC3)=O)cnn12 36820,C1(NC(=O)Cc2ccn(C(F)F)n2)CCC(CNC(C2(Cl)CC2(F)F)=O)CC1 36821,c1(NC(N2CCOCCC2c2ccc(F)cc2)C)ccc(S(=O)(=O)C(C)C)cc1 36822,c1(C(=O)NC2(CCCNC(COCCOC)=O)CC2)cnc(N)c(O)c1 36823,N1(C(c2c(CCCC)ocn2)=O)CCN(C(=O)Cc2ccns2)CC1CO 36824,C(C(C)(C)C(=O)NCC)NC(CC1C(CNC(C2N(CC)CC2)=O)C1)=O 36825,Cc1c(C(=O)NC(C2CCCN2C(=O)Cc2cn(C)nc2Cl)C)sc2nccn12 36826,c1(C(N2C(COC)CN(C(c3nc(Cl)sc3C)=O)CC2)=O)cc(C)cc(C)c1O 36827,O(C=CC(=O)N1CCCC1C1CCN(C(=O)C(F)CN(CC)CC)C1)CC 36828,c1(NC(C2N(C(c3c(COC)onc3)=O)C3C(C2)C3)=O)ccc(C#N)cc1C 36829,C(=O)(CC1CCC(C)(C)c2ccccc21)NCCCNC(C(COC)O)=O 36830,CN=c1[nH]ccc(C(N2CCCC(NC(C3(F)CC=CCC3)=O)C2)=O)c1[N+](=O)[O-] 36831,c1(SC)ncc(C#N)c(N2CCCC(C(N3CCCC(CO)C3)=O)C2)n1 36832,c1(NC(CC2N(C(C(C3CCCCC3)OC)=O)CC2)=O)ccc(C)c(C2CC2)c1 36833,c1(CC)n[nH]cc1C(=O)NCCOCC(N1CCC(NC(C)=O)C1)=O 36834,C(CC(C)C)(C(=O)N1CCC(C)C(C(=O)NOC(COC)COC)C1)OC 36835,C=CCC(C(=O)N(C(C)C(F)F)C1CC1)NC(=O)C(C)NC=O 36836,N1(C(=O)CC2CC=CC2)CC2(CCN2C(c2cc(-c3ccncc3)on2)=O)C1 36837,C1(CC(N2CC(CNC(Cc3cccc(SC)c3)=O)C2)=O)CCC2(CCC2)CO1 36838,CCCC(CCNC(=O)C(C)(C1CCC1)NC(=O)CSC(C)(C)C)C1CC1 36839,Cc1cc(O)ccc1C(=O)NCC1CCCN(C(=O)CCC2CCCN2C)CC1 36840,Cc1nn(CC(F)F)c(C)c1C(=O)NC(C)CCCNc1ncncc1Cl 36841,CC(CC(F)F)C(=O)N(C)CC1CCCCN1C(=O)C(O)Cc1ccccc1 36842,N1(C(C2CC(=O)NCC2)=O)CCC(CNC(=O)CCc2ncc[nH]2)C(F)(F)C1 36843,c1(CNC(C2C(CNC(=O)CC3CCCOC3)CCC2)=O)ccnc(O)c1 36844,Cc1nc(CO)sc1C(=O)NC1(C)CCN(C(=O)CSCc2csc(=N)[nH]2)C1 36845,C1(C(=O)NC2CC3(C(NC(c4ccc(CC)cn4)=O)C3)C2)CCc2nc[nH]c2C1 36846,N1(C(C2CCC(=O)O2)=O)CC2(C1)CN(C(c1cccc(C(F)F)n1)=O)C2 36847,N1(C(C(CC)NC(C)=O)=O)CCN(C(=O)Cc2nc([N+](=O)[O-])n[nH]2)C(C(C)C)C1 36848,c1(-n2c(C(C(C(C)C)OC)NCCCC=C(C)C)nnn2)ccc(F)cc1 36849,C1(CN(C(=O)CC2CC3CC3C2)CC)CCN(C(C2(SCC)CCCO2)=O)CC1 36850,C1(C(=O)NCC2CCC(F)(F)CC2)CC2CCC1N2C(c1cccc(=O)n1O)=O 36851,N1(C(C2(C)CC(=O)C2)=O)CCC(C)(C)C(CNC(c2c(F)cccc2F)=O)C1 36852,N1(C(CCNC(CC(CC)C2CC2)=O)=O)CC2CCC(C1)O2 36853,N1(CCC)CCN(S(=O)(=O)N(C)C)CC1.c1(C2CNC(=O)N2)c(F)cccc1F 36854,N1(C(C(CC)NC(C)=O)=O)CC=C(CCNC(C2C(C)OC(C)C2C)=O)CC1 36855,c1(CC(=O)NC2CCCCCC2NC(=O)CC(F)(F)F)cccc2c1OCCC2 36856,C1(C(N(C)CC2CCN(C(c3ccoc3C3CC3)=O)C2)=O)CCC(C)(C)CC1 36857,C1(CN)CCN(C(=O)Cn2cc(CN3CCCCC3)nn2)C1 36858,CC(C)CC(C)CC(=O)N1CCC1CNC(=O)CCc1nncn1C 36859,N1(C(c2c(C)nc(CC)s2)=O)CC2(CCCCN(C(C3CCCCC3C)=O)C2)C1 36860,C1(NC(CSc2c(C)n[nH]c2C)=O)CCN(C(c2nccc(CO)n2)=O)C1(C)C 36861,c1(N(C)CCOCC(C)(C)C(C)(F)F)ccc(S(=O)(=O)NC2CC2)cn1 36862,N1(c2nccc(CC)n2)CCC2(NC(c3cn(C)nc3COC)=O)CCCC12 36863,c1(CC)cc(Cl)ccc1NC(c1nnnn1C1CCOCC1)CC1COC1 36864,c1(-c2nc(C)c(C(=O)Nc3cc(F)c(Cl)cc3F)cc2)ccc2c(C)[nH]nc2c1 36865,c1(OC)cc(SC)ccc1CNC(CN(C)C)CC(C)C 36866,C1(CC)CCC(CNC(=O)C=CC(C)(C)NC(=O)Cc2ccn(C)c2)CC1 36867,C1(OCCCCOC(c2cn(C3(C(=O)O)CC3)nn2)=O)C=CCCCC1 36868,C1(NC(CSCC=C)=O)CC(OC)CN(C(=O)CCc2cc(C)nc(C)c2)C1 36869,c1(C(N2CCCC(F)(CNC(C3C(C)(C)CC3)=O)C2)=O)n[nH]c2cc(Cl)ccc12 36870,N1(C(CCCCCOC)=O)CC2CCCN(C(=O)CCC(C)(C)C)C(C2)C1 36871,C1(NC(c2cccc(C)n2)=O)CC2CC1N(C(=O)C(F)(F)CCn1ccnn1)C2 36872,C12CCC(O1)C(C(=O)OC)N2.c1(CCNC(=O)OC(C)(C)C)csc(=N)[nH]1 36873,C=C(C)C(CC(=O)N1CC(OC(=S)NC2CCCCC2)C1)OCc1ccccc1C 36874,c1(OCC)ncc(NC(=O)C(C2CCCN(C(=O)C(C)C(C)C)C2)(C)C)cn1 36875,CC(C)CC(F)(F)C(=O)NC1CN(C(c2c(Cl)nn(C)c2Cl)=O)CC2(CC2)C1 36876,C(=O)(CC(C)CC(=O)NCCC(C)NC(=O)Cc1ncn2c1CCCC2)OC 36877,N12CCCC(C1C)N2C1(C)CCN(C)CC1.c1(C(=O)OC)ccn(O)c(=O)c1.SC 36878,N1(C(c2cn(C3CC3)cn2)=O)CCCC(F)(C(N2CCCCC2CO)=O)C1 36879,c1(C(N2CCC(N(C(c3c[nH]nc3SC)=O)CC)C2)=O)cn2ccc(C)cc2n1 36880,C1(C(=O)NC(CNC(C2CC(OCC)C2)=O)C2CCC2)CC(O)(C(F)(F)F)C1 36881,C1(C(=O)NC(c2nccs2)C)CCCC12CCN(C(c1ccc[nH]1)=O)C2 36882,c1(C(N2CC(C)C(CNC(c3cn[nH]c3)=O)C2)=O)nc(Br)c2ccccn12 36883,N1(C(C(C)C)=O)CCN(C(=O)C(O)CCN(C)C)C(C2CC2)C1 36884,Cc1ccc(C(=O)N(C2CCCC2)CCNC(=O)C(C)(C)C(N)=O)c(C)c1Br 36885,c1(C(c2nnnn2C2COC2)NC(C2COC2)C)c(Br)nc2n1CCOC2 36886,C(=O)(C(F)CC1CN(C(C2CC2c2ccccc2)=O)C1)N(C(C)C)C1CC1 36887,C12(CNC(=O)COc3ccon3)COCCN1C(=O)CN(C(C1CCOC1)=O)C2 36888,c1(C(N2CC(O)(CN(C)C(c3cccn3C)=O)C2)=O)cccc(F)c1F 36889,CC1CN(Cc2ccccc2)CCC1NCc1ccnc(C2CCCC2)n1 36890,N1(C(C(c2ccnn2C)C)=O)CCC=CC1C(N1CCC1CF)=O 36891,C1(NC(=O)CCc2ccccc2Cl)CC2CC1CN(C(=O)CC1CC(F)C1)C2 36892,c1(NC(C2(NC(CCOCC)=O)CCCC2C)=O)c(C)ccn(C)c1=O 36893,c1(C(N2CC3CCC2CN3C(C23CCC2C3)=O)=O)cc2oc(Br)cc2[nH]1 36894,CCC(C)CC(=O)N1CCC(O)(CCNC(C2CCCC2OC)=O)C1 36895,c1(C(N2C(C(=O)NC(COC)C)CC(F)C2)=O)cc(Br)ccc1C(F)(F)F 36896,c1(CCCC(=O)NCC(CC=C)NC(C2(COC(C)C)CC2)=O)ccc(O)cc1 36897,c1(C(=O)NC2CC(=C)CN2c2nccc(C(=O)OC)n2)cc2sccc2s1 36898,N1(C(C(CC)N(CCO)CC)=O)CC2(CC(C(=O)NOC3CCCCC3)CO2)C1 36899,S(=O)(=O)(c1cnc(NCC2(Br)CC2)c(Cl)c1)N1CCCC(C(C)O)C1 36900,CC1(C)CN(C(C2CCN(C(C3CC(O)C3)=O)C2)=O)CC1O 36901,C(C(=O)NC(C)(CNC(=O)C=Cc1cn[nH]c1)CO)(C(C)(C)C)SC 36902,c1(CC(=O)OCC)ncc(NC(=O)C(C(C)C)NC(=O)CC(C)C)cn1 36903,C12(C(N(C)CC3CC(O)C3)=O)C(NC(C3CC4C=CC3O4)=O)C3CC1C2C3 36904,c1(CC(=O)NC(CNC(Cc2c(C)nsc2)=O)(C)C)cccc(OC(F)F)c1 36905,C1(CNC(Cc2cc(OC)ncc2)=O)CCN(C(C2CC=C(C)CC2)=O)C12CC2 36906,C12(CC)CCC(C(=O)NC3CCC(NC(C4(C)CC(F)C4)=O)C3)(CC1)CO2 36907,N(C(=NCC1CCC1)N1Cc2ccccc2C(F)(F)C1)Cc1c(OC)ccnc1 36908,N1(C(c2c(N)ncc(C)c2)=O)CC2CC3CC2C1C3NC(c1csc(C)c1C)=O 36909,c1(C(=O)NCCCC(C)NC(CCCCC)=O)ccccc1C#N 36910,CC1CN(C(=O)C(C)(C)C2CCN(C(C3CC(F)CN3C)=O)C2)CC1O 36911,O=C(CC1CCNCC1(F)F)NNc1nc2ccccc2s1 36912,N1(C(c2sc(C(F)F)nc2Br)C(=O)NCCCC)CC2(CCC2)CC1CO 36913,C(C(C)(C)C#CC(=O)NCC(O)CC(F)(F)F)NC(C(C1CCCCCC1)C)=O 36914,C1(C(N(CCOC)CCO)=O)CCN(C(C2(CO)CCCCO2)=O)CC1(C)C 36915,C1(NC(C2(C(=O)OCC)CCCO2)=O)CCC(C#N)CC1 36916,Cc1c[nH]nc1C(=O)N(CCCNC(=O)C(Cc1ccccc1)N(C)C)C 36917,C1(OCC)CN(C(c2nccc(C)n2)=O)CC1CNC(c1ccc(SC)cc1)=O 36918,C(CCCC(=O)N1CCC(N(C(=O)C(c2nc(C)cs2)C)C)C1)(OC)OC 36919,N1(C(C(CC)N(C)C)=O)CCSCC1CCNC(=O)C(O)c1ccco1 36920,C(=O)(C1CCC(=O)c2cccn21)NCCC1(O)CN(C(c2cnn(C)c2F)=O)C1 36921,c1(C(=O)NC2CN(C(C(C)C)=O)CC23CCC3)nn(C)c2ccccc12 36922,c1(C(=O)NCC2CC3CN(C(C4(C)CC4(F)F)=O)CC32)cc2ncccc2[nH]1 36923,c1(CNC(C2(CCC)CCC2)=O)cc(C(=O)NCCCCCF)co1 36924,c1(C(N(C)CC2CCN(C(CCSCC)=O)C2)=O)cccc(-n2ccnc2O)c1 36925,C1(OC)CC(NC(c2cc(C)nc(O)c2)=O)CN(C(=O)C(C)Cc2cnc[nH]2)C1 36926,C(=O)(CC(O)C(C)C)NC1C(NC(C(CC#C)C)=O)CCCC1 36927,N1(C(C2(SC)CC2)=O)CC(CCC(=O)NC2(CC(C)C)CC2)C1 36928,N1(C(c2ccn(CC)n2)=O)C2CCC(C2)C1CNC(c1cc(C)c(C)o1)=O 36929,C(=O)(CC(F)(F)F)N.C1(CCNC(C2CCC(C(F)(F)F)C2)=O)(OC)CN(C=O)C1 36930,c1(C(N2C(C)CCC(NC(C3CCN(C)S3(=O)=O)=O)C2)=O)ccc2cncn2c1 36931,Cc1c(N)cc(C(=O)NCC(C)NC(=O)C(c2cccc(Cl)c2)O)cc1[N+](=O)[O-] 36932,c1(C(N2C(CNC(c3n(CCC)ncc3)=O)CC2)=O)cc(C2CC2)nc2ccnn12 36933,C1(N(C)C)CN(C(C23CC2CCN3C(C2CC(N(C)C)C2)=O)=O)CC1(C)C 36934,N1(C(C(CNC(C2C=C(C)CS2)=O)OC)=O)CCOC(C)(C)C1C 36935,c1(CNC(C2(CCC)CC2)=O)ncoc1CCNC(C1CC(C)(C)O1)=O 36936,Cc1cc(O)ccc1C(N1CC=CC(NC(=O)Cn2cccnc2=O)C1)=O 36937,c1(C(=O)NC2C3(CC(NC(c4c(C)cc(Br)o4)=O)C3)C2)cc[nH]c2nccc1-2 36938,C(=O)(CCC(=O)OCc1csnc1C1CC1)OCC 36939,c1(CC(N2CCC(C(C)NC(=O)C(N)=O)C2)=O)cccc2ncccc12 36940,C(=O)(C(C)(C)CCCNC(=O)C(c1cnn(C)c1)C)N1C(CC)CCOCC1 36941,C(C(C)(Cn1cccn1)NC(c1c[nH]c(=N)o1)=O)NC(CSC)=O 36942,c1(C(N2CCC(NC(C(CCSC)OC)=O)C(F)C2)=O)cc2oc(C)c(C)c2[nH]1 36943,c1(CC(=O)NC2(C)CCCO2)cccc(OCc2ccccc2O)c1 36944,CC1CCN(C(=O)C(c2ccoc2)NC(=O)COCCC(C)C)CC(C)O1 36945,CCCC(C)(C)C(=O)NC1C=CC(C(N2CC(=O)NC(C(=O)OC)C2)=O)C1 36946,N1(C(c2cnc(OC)c(Cl)c2)=O)CC(F)(F)CC1(C)CNC(C1CCSC1)=O 36947,CC1(c2ccc(-c3noc(CCNC(=O)OC(C)(C)C)n3)cc2)NC(=O)NC1=O 36948,c1(C(C(=O)NCC2CCOC2)N(C)Cc2cnc(CC)s2)ccc(C)cc1Cl 36949,C1(C)(CC)C=C(C(=O)N2CCOC(CC(=O)NCCOCC(C)(C)O)C2)C1 36950,C(=O)(C(CO)C(C)(C)C)NC(CCC#C)C(=O)NC(c1ncc(C)cn1)C 36951,C(=O)(C1CCc2c[nH]nc21)N1CC2(C(NC(=O)Cn3ncc(O)nc3=O)CC2)C1 36952,c1(C(=O)NC2CCCN(C(CC3(COC)CC3)=O)C2)cc2cc(F)cc(F)c2[nH]1 36953,C1(=CC(=O)NC2(CC=C)CN(C(c3ccc(CSCC)o3)=O)C2)CCC(C)CC1 36954,C1(O)(C(C)(C)OC)CC(NCCN(c2ccccc2)S(C)(=O)=O)C1 36955,C1(O)(CNC(C(C)=C2CCCC2)=O)CCN(C(=O)C(O)C2CCCC2)CC1 36956,CC(=O)C(C)(C)CC(=O)N1CC=CC(C(=O)NCC=CCCOC)C1 36957,CCC(C)CCN=c1[nH]c(=NCC2(COC)CCC2)c2ncccc2[nH]1 36958,CC1(C(=O)NCC(C2CCN(C(C3CC4(CC4)CO3)=O)CC2)O)CCC2CC2C1 36959,c12cccc3c1CCN(CC3)C2.C1(OC(C)=O)CCSCC1 36960,c1(CC2(C(N)=O)CCC2)ccc(OCC(=O)NCC2(NC(=O)C3CC3)CC2)nc1 36961,C(=O)(C1=COCCC1)N(CCNC(CS(CC)=O)=O)CCc1ccccc1 36962,C1(C(=O)NCCC2C(C(=O)OC)C2)CN(C(C2COCCC2C)=O)CC1F 36963,Cc1cc(C2(C(=O)N(C3CCCN(C(C4CC4(Cl)Cl)=O)C3)C)CC2)cc(C)c1 36964,Cc1ccnc(-n2cc(CN3CCC(C(NOCCCC(F)(F)F)=O)C3)nn2)n1 36965,c1(C(=O)NCCC2(O)CN(C(CC=C(C)C)=O)C2)cnc(N(C)C)nc1 36966,N1(C(COCCC=C)=O)CCCC(O)(CNC(=O)C(C(C)C)SCC)C1 36967,N1(C(CCCCC(N)=O)=O)CC(NC(c2cccnc2)=O)CC12CCCOC2 36968,C(CN=C(NCc1cccc2c1OC(F)(F)O2)N1CC(O)C(C)(C)C1)SC 36969,c1(C(=O)NC2(CCNC(CSCCC)=O)CCC2)scc(C)c1C 36970,CCCCC(O)C(=O)N(CC(=O)NC1(CC)CCCC1)C(C)C 36971,C=C(C)c1cncc(C(c2nnnn2CCCSC)NCC2(C#N)CCCC2)c1 36972,C(=O)(C#CC1(C)CCCO1)N(CCC(=O)NCC(CC)C(C)C)C(C)C 36973,c1(NC(COC2CN(C(c3cncn(C)c3=O)=O)C2)=O)cn(C)c(=O)nc1O 36974,c1(CN(C(C(CNC)(C)C)=O)C(C)C)cc(OC)c(OC)c(OC)c1 36975,C1(O)(CC)CCN(C(=O)C=CC(C)NC(C2CCCC2O)=O)C1 36976,N1(C(c2ccn(CCCC)n2)=O)CCC2(NC(=O)C=CC3CC3)CCCCC12 36977,c1(OC)ccc(F)c(C(=O)NCC(C2CCC2)NC(C23CC(OC)C2C3)=O)c1 36978,C1(CNC(CCOCCC)=O)CCC2(CCC2)CN1C(=O)C(C)C(C)COC 36979,c1(OCCCC(N2CC(O)(CNC(c3cc(CC)on3)=O)C2)=O)ccc(Cl)cc1 36980,C=CCC(CC=C)C(=O)N1CCC(C(=O)N(CCCCC)C)(CC)C1 36981,C1(NC(C(C)(C)OC)=O)CCC(C)C(C)C1 36982,c1(C(=O)NCC2C(C)CCN(C(C3(CC=C)CCC3)=O)C2)cnc2c[nH]nc2c1 36983,N1(C(C(C)S)=O)CC(Oc2ccccc2)CC1CNC(C1CCSCC1)=O 36984,n1(CC(=O)NC2CC2)ccc(=NC(=O)CSc2cccc(C)c2OC)nc1O 36985,c1(C(=O)NCC2N(C(C(CC)C)=O)CC(C(F)(F)F)C2)cncc(F)c1C 36986,c1(C(N(C2CCC(NC(=O)C=CCN(C)C)C2)C)=O)ccc(OC(F)F)nc1Cl 36987,CCCC(C)(CC)C(=O)NCC1(OC)CN(C(C23CCCC2C3(F)F)=O)C1 36988,C1(C(N(C2CN(C(C(c3cccnc3)C)=O)C2)C)=O)C(C)(C)C1(C)C 36989,C1(NC(C=C(C)C(C)C)=O)CC2CN(C(=O)CN3CCCCC3=O)CCN2C1=O 36990,CCC(CC)C(=O)NCC.C1(C)CC(CNC(=O)COCCOCCOCC)CO1 36991,c1(-c2nc(C(C)Nc3cc(S(C)(=O)=O)co3)[nH]n2)ccc2ccccc2c1 36992,c1(CC(=O)NCC2C(C)CCCC2)cc(Br)ccc1Cl 36993,Cc1cc(C(=O)NCCCCC(C)NC(=O)CCC2(C)CC2)cc(N)c1 36994,N1(C(C(C)(C)OC)=O)CCC(CC(=O)NC(C)CC2CC2)CC1 36995,c1(CNC(C2CCN2C(=O)OC(C)(C)C)C)ncc(Cl)cc1Cl 36996,c1(OC)c(CN2CCSC(C(=O)Nc3cnc(Cl)nc3C)C2)cc(Cl)cc1Cl 36997,N1(C(C2(CCC)CC2)=O)CCC2CCCN(C(c3cn(C)nc3C)=O)C2C1 36998,C1(NC(C=NOC)=O)C2CCN(C(=O)C(C)Cc3cccnc3)CC12 36999,C1(C(=O)NCC2N(C(c3nc(C)sc3)=O)CCCC2)CC2CC1C1C2C1(F)F 37000,C#CCC(CC(F)F)C(=O)N1C(C(=O)NCC2(O)CCCCC2)CCC1C1CC1 37001,c1(C(C)C)cc(C(=O)NCC2CN(C(=O)CCSC(F)(F)F)C3CC23)ccc1F 37002,c1(C(=O)NC(C2N(C(c3c(C(C)C)ncs3)=O)CCC2)C)cc2n(n1)CCC2 37003,c1(OC)ccc(Br)c(C(N2CCCC(O)(CNC(=O)C(C)SC)C2)=O)c1 37004,c1(C(=O)NC2C(NC(C(CC)O)=O)C2)ccc(C(F)F)nc1 37005,C1(OCC)CC(NC(=NCCF)NCC2CCSCC2)C12CCCCC2 37006,C1(C(=O)NC(C)C(CO)NC(=O)Cc2ccn(C)c2)(COC)CCCC1 37007,c1(C(=O)NC(C2CCOC2)CC)ccc(Cn2cc(C(N3CCCC3)C)nn2)o1 37008,c1(CNC(NCc2n(C)ncc2Cl)=NCC2CC2)ccccc1N=[N+]=[N-] 37009,c1(N2CCC(c3onc(-c4nccc(C)c4)n3)C2)cc(Cl)ccc1Cl 37010,C1(NC(C(F)=C(C)C)=O)CCCC(NC(c2cc(Cl)n(C)n2)=O)C1 37011,c1(C(N2CC3CC2CN3C(c2nc3ccccc3o2)=O)=O)cccn2ncnc12 37012,CC1CCC(O)(C(=O)NC2CCCN(C(=O)C(C)CSC(F)(F)F)C2C)CC1 37013,C1(C2CCN(C(=O)CCc3cc(F)cc(F)c3)C2)(NC(C2C(C(C)C)C2)=O)CC1 37014,c1(C(=O)NCC(CN(C(C2(OCC)CCC2)=O)C)O)c(C)nn(C)c1N 37015,CC(C)C(CC(=O)N1CCC(O)CC1)NC(c1cocn1)=O 37016,CCC(CC(=O)NC(C(=O)NCCC1(COC)CCC1)C(C)O)OC 37017,CC(C)C1=NOC(C(=O)NCC2CC3CCC2N3C(C23CC(C)(CO2)C3)=O)C1 37018,CCC(C)C(O)C(=O)N1CCCN(C(c2[nH]c(-c3cccnc3)nc2C)=O)CC1 37019,c1(C(=O)NCCC(C)NC(c2cnnn2C)=O)c(Cl)c(Cl)cc(Cl)c1Cl 37020,c1(C(=O)NC(C)Cn2cc(Br)cn2)cc(S(=O)(=O)N(C)C)ccc1Cl 37021,N1(C(c2ccc(C)n2C)=O)CCCCC2(CCN(C(c3cncc(N)n3)=O)C2)C1 37022,CC1(C)CCCCCC1NCC1CCCNC1 37023,Cc1ccc(I)c(C(=O)NC2CN(C(=O)Cc3ccc(F)cc3F)CC23CC3)c1 37024,C1(N(N2CC(c3cccc(C(N)CCCC)c3)C2)C2CCCO2)CCNC(=O)CC1 37025,CP(C)(=O)C(O)C(=O)NC1CCCN(C(c2ccc(OC(F)(F)F)cn2)=O)CC1 37026,CC1CNc2cc(C(=O)NC3CCC(NC(C4CC(F)C4)=O)CC3)ccc2O1 37027,C(C(C(=O)NOCCCC(=O)OC)C(C)(C)C)NC(C(CCC)C#N)=O 37028,N1(C(c2cc(OC)n[nH]2)=O)CC(CNC(C2CCCN2C)=O)C2(CC2)C1 37029,C1(C(=O)NCCCCN2CCOC2=O)Cc2ccc(Br)cc2N1 37030,c1(N2CC3CN(C(Cc4cc(C)cc(C)c4)=O)CC3C2)nc2ccc(Cl)cc2s1 37031,C=C(C)C(CC(=O)NCC1CCC1NC(=O)Cc1ccc(F)cc1F)OOCC 37032,C1(NC(C2CCCC(F)(F)CC2)=O)CCN(C(c2n[nH]cc2F)=O)CC12CCC2 37033,C1(C(=O)NCC=CCCC)(C(C)C)CCN(C(=O)CCC=C(C)C)C1 37034,c1(C(=O)NC2CCCC(N(C(=O)C#CC3CCC3)C)C2)cc2ccccn2n1 37035,C1(NC(CC=CC)=O)C(CNC(=O)COc2c(C)cccc2Cl)CCC12CCC2 37036,C1(CC(=O)NCCOC2CCN(C(C(C)(C)CC3CC3)=O)C2)CCCCC(=O)N1 37037,Cc1nn[nH]c1C(N1CCCC1CCNC(=O)CC1(CS(C)(=O)=O)CC1)=O 37038,c1(C(=O)NC2CS(=O)(=O)CC2NC(c2cnccc2Cl)=O)cn2cnnc2cn1 37039,C12(C(=O)NC3CC(NC(C(CC)(C)O)=O)CC3O)CC3CC(C(=O)N1)C2C3 37040,c1(OC)c(C(=O)NCC2CCCN(C(=O)C(C)S(N)(=O)=O)C2)ccc(Cl)c1C 37041,N1(C(C2N(C(C(C)NC=O)=O)CC(F)C2)=O)CCOC(C)(C)C1 37042,c1(C(N(C)CC2CN(C(c3ccncn3)=O)C2)=O)cc(N)cc(O)n1 37043,C1(C(N(CCOCCNC(c2c(C(C)C)scc2)=O)C)=O)CC2CCCC2C1 37044,C1(=O)C(C)(C)CC(=O)NCCCN1CCC.N1(C(C)=O)CCOCC(C)(C)C1 37045,N1(C(CC(CC)CN(C)C)=O)CC2CCCC(C1)N2C(=O)C1=NNC(=O)C1 37046,N1(C(c2c(C)cccc2)=O)C2CCC1(CNC(=O)CCCC(=O)NC(C)C)CC2 37047,c1(NC(=O)NCC(C)(CC2CCCC2)NC(=O)OC(C)(C)C)cnccc1C 37048,C1(CC(=O)N(CC(N2CC(C(N)=O)(N(C)C)C2)=O)C)CCCC1O 37049,CC(C)CC(CNC(C1(C(F)(F)F)CC(F)(F)C1)=O)NC(c1ccccn1)=O 37050,C1(CC=CC)CCCN(C(=O)CC2CC2CNC(=O)C(C)SCC)C1 37051,C1(NC(c2c(OC)cnc(Br)c2)=O)CC2(CCN(C(c3ccccc3)=O)CC2)C1 37052,N1(C(CC(COC)C)=O)CC(NC(c2cccc(C(F)(F)F)n2)=O)CC12CCC2 37053,c1(OC)cnn2c1CN(C(=O)Cc1ccc(-c3nn[nH]n3)cn1)CC2 37054,C1(C(=O)NC23CC(NC(c4c(CC)c[nH]c4)=O)(C2)C3)CC(=O)NC(C)C1 37055,c1(CC(C)CN2CCCC2)cc(C(=O)O)cc(Cl)c1 37056,CC1CN(CC(=O)NCC2CCN2C(C2CC2C(c2ccccc2)=O)=O)CC1 37057,Cc1cc(F)ncc1C(=O)NC(C)CC1CN(C(=O)CCOC2CCOCC2)C1 37058,N1(C(c2cc(COC)[nH]n2)=O)CC2CCC(C1)C2NC(c1cc(COC)cs1)=O 37059,c1(NC(N2CCC(CCC=C)C2)=O)c(I)cnc(Cl)c1F 37060,c1(C(=O)OC)cc(NC(C2C(C(=O)NCC3(c4cc[nH]n4)CC3)C2(F)F)=O)on1.OC 37061,c1(C(CC(=O)NC2CN(C(C3(C(=O)OCC)CC3)=O)CC2O)C)ccc(F)cc1F 37062,N1(C(=O)C=CCN2CCCC2)CC2(C=C(C(=O)NCc3[nH]nnc3CO)CO2)C1 37063,c1(-c2cc(C)cc(O)c2)ccn2cc(C(=O)NCC(F)F)nc2c1 37064,N1(C(CN(C)C)=O)CC2CCCN(C(c3ccc4oc(O)nc4n3)=O)C2C1 37065,Cc1ccc(OCC(=O)NC2CCC23CN(C(c2[nH]ncc2C#N)=O)C3)c(C)c1 37066,c1(C(=O)NCC(CNC(C(C)SCC)=O)F)cc(F)cc2nn(C)cc12 37067,Cc1cccc(C(=O)NC2CCC(C)(CNC(c3cc(C(F)(F)F)no3)=O)C2)n1 37068,c1(C(CC)CC)cc(C(=O)NC2CC(CNC(=O)CN3CSCC3=O)C2)on1 37069,C=CC(CC)CC(=O)NCCN(C(=O)C(C)(C)F)Cc1cccc(Cl)c1 37070,c1(C(N2CC(CNC(C=CC(=O)OCCCC)=O)C2)=O)cc(N(C)C)ccc1F 37071,c1(C(=O)NCCC(C(C)C)NC(c2nc(C)sc2)=O)c[nH]c2cc(F)ccc12 37072,c1(C(=O)NC2CN(C(C3(C=C)CCCCC3)=O)CC(C)C2)cc2ncccc2o1 37073,C1(NC(C2C(C)(C)CCC2)=O)CCC(O)CN(C(=O)C2=CCCSC2)C1 37074,c1(C(=O)NC2CCC(NC(c3c(SCC)nccn3)=O)C2)cc(CC)ccc1O 37075,N1(C(C2CC23CC3)=O)CC2(C(=O)NCCOCCF)CCC1CC2 37076,c1(C(N(CCC(=O)NCC2NC(=O)NC2=O)CC#C)=O)cccc(CC=C)c1 37077,c1(C(=O)NCC2COCC2NC(C2(C(F)F)CC2)=O)cn2cc[nH]c(=O)c2n1 37078,n1(C(C)C(N2CCOCC2)=O)cc(CN(C2CCOCC2)C)nn1 37079,C(=O)(C1=C(C)OCC1)N(CCCNC(c1cnc(F)s1)=O)CC 37080,c1(C(=O)NCC(=O)NC2C(CNC(=O)CCn3cncn3)C2)ccc(Cl)cc1Cl 37081,Cn1ccc(C2(C(N3CC(O)(CNC(c4csc(C(F)F)c4)=O)C3)=O)CC2)n1 37082,c1(NC(C2CC3CCCCC3N2C(c2ccoc2)=O)=O)ccc2nc(O)[nH]c2c1 37083,N1(C(C2CN(C(N)=O)C2)=O)CCC(CC(c2ccccc2)O)C1 37084,N1(C(C2N(C(C)=O)CCC2)=O)CCCCCC(NC(c2csc3cncn23)=O)C1 37085,c1(C(=O)NC2CCN(C(C3CC(CC)(CC)C3)=O)C2)cc(C)c(Cl)cc1OC 37086,N1(C(CC2CC(OC)C2)=O)CCCC(C)C1CCNC(=O)CCC1CC(F)(F)C1 37087,C(=O)(CCCN=[N+]=[N-])NC1C(NC(c2nn(C(CC)C)c(C)c2)=O)COCC1 37088,N1(C(c2c(CC)non2)=O)CCC(CN(C(=O)CC2(COC)CC2)C)CC1 37089,c1(N2CCC3(CC(OC)C3)C2)nc(=NCc2cc(C)cs2)[nH]c2c1CCC2 37090,N1(C(C(C)OCC=C)=O)CC2CCCC(NC(c3cc(O)cc(=O)o3)=O)(C2)C1 37091,c1(NC(c2c(CC)ncs2)=O)ccc(C)c(C(F)(F)F)c1 37092,C12CC3(C1)CC3N2.n1(NC(=O)CCc2ccc(C3CC3C)o2)ccc(CC)n1 37093,c1(C(=O)NCCC2CC(NC(c3cn(CCO)nn3)=O)C2)cc(Cl)ccc1O 37094,C1(CC=C)(NC(C2CC3CC3C2)=O)CCCN(C(C2CC(=O)N(C3CC3)C2)=O)C1 37095,C1(NC(Cc2c(C)n[nH]c2C)=O)CCCN(C(=O)CNC=O)CC1F 37096,c1(CC(C(=O)NC2CCC(NC(CCSCCC)=O)CC2)C)ccc(F)c(F)c1 37097,CCCCCCC(C)(CC)C(=O)Nc1ncc(Br)c(C)n1 37098,C1(C)(C(c2n(CCSC)nnn2)NCCC(=O)NC(N)=O)CCOCC1 37099,C(C(C)(C)CNC(c1nonc1N)=O)N(C)C(C1C=CCCC1)=O 37100,C1(CN(C(=O)CC2CC(C)(C)C2)C)C2CN(C(=O)CC(C)(F)F)CC12 37101,C(=O)(C1=CC2C=CC(C1)C2)NC(CC(CC)C)C(=O)N1CCC12CC(CN(C)C)C2 37102,c1(C(N2C(C(=O)Nc3c(C#N)cnn3CCO)CC2)=O)ccccc1[N+](=O)[O-] 37103,c1(SC)ccccc1C(=O)NC(C1CN(C(=O)Cc2cncc(O)c2)CCO1)C 37104,C(=O)(C1=CS(=O)CCC1)N1C(CNC(C=Cc2c(C)ccs2)=O)COCC1 37105,c1(OC)nccc(=NC2CCCOC3(CCCOC3)C2)[nH]1 37106,c1(N(CC(=O)NCC(CCCC)NC(=O)CC(F)(F)F)C)ncnc2[nH]cnc12 37107,Cc1ccc2oc(C(=O)NC3CN(C(=O)CCNC(=O)CO)C4CC34)cc2n1 37108,C(=O)(C(=O)C(C)(C)C)N1CCC(OC)(CNC(c2ccccc2SC)=O)C1 37109,CC(C)CC(C)(CNC(C1(C(C)(F)F)CCC1)=O)NC(c1cnc2n1CCC2)=O 37110,C1(NC(CC)=O)CCCC(N(C(=O)C#CC(C)NC(=O)OC(C)(C)C)C)C1 37111,c1(NC(N)=O)cc(Br)cnc1N1CCCC(Cc2ccc(Cl)cc2)C1 37112,CCC(C)(C(=O)NC(CNC(=O)C=Cc1cccc(F)c1F)C(C)C)C(F)F 37113,C(=O)(C(CC)C(C)O)N(CC(CC1CN(C(C(CC)CC)=O)C1)(C)C)CC(C)(C)C 37114,c1(C(C)N)ccc(Oc2ccc(CNC(=O)CCC3CCC(=O)NC3)cn2)cc1 37115,N1(C(C2CC(N(C)CC)C2)=O)CCC2CC12C(=O)NCCC12CCC(CO1)C2 37116,N1(C(C(N2CCC(C)CC2)=O)=O)C(CNC(=O)C=CC2CCC2)CC2CCCC12 37117,c1(OC(CC)C(=O)NC2CCCN(C(=O)C=CBr)C2)ccccc1F 37118,C1(NC)CCC(C(=O)N(CCC(=O)NCC2CCCC2)CCO)C1 37119,C(=O)(C(O)P(C)(C)=O)N1CCC(N(C(CSS(C)(=O)=O)=O)CCO)C1 37120,C1(OC)CC(CO)N(C(c2csc(NC(C3CC3C3CCN(C)CC3)=O)n2)=O)C1 37121,c1(C(c2n(C(CC)C)nnn2)NCCCOC2CC2)nc(C)c(C)n1C 37122,c1(CCC(=O)N(CCCNC(C2CCC2C(F)(F)F)=O)CC)nc(C(C)C)no1 37123,C1(c2nnnn2C)(Nc2c(NCC)c(CC)ccc2)CN2CCCC2C1 37124,CCC(C(=O)NC1CC1NC(=O)CCc1sccc1Br)c1ccccc1 37125,Cc1cnc(C(=O)NCC2C(C)CCN2C(c2cc(C3CC3)nn2C)=O)cc1C 37126,c1(OC)ccc([N+](=O)[O-])cc1C(N1CCC12CN(c1ncccn1)C2)=O 37127,c1(OCC(=O)NC(CC)CNC(C2CC23CC3)=O)ccccc1OC 37128,N1(C(C(Br)=C(C)C)=O)CC(C)OC2(CCN(c3ncc([N+](=O)[O-])cc3Br)C2)C1 37129,CCCCC(C(=O)NC1CCN(C(C2CCCCS2)=O)C1C(C)C)N(C)C 37130,N1(C(C(C)SC(F)(F)F)=O)CC(CO)C2(C1)CN(c1ncnc3c1cnn3C)C2 37131,C1(CNC(C2CN(CC)C(=O)C2)=O)C(C)CCCN1C(=O)Cc1ccc(Cl)s1 37132,c1(NCCOCCNC(C2CC3CCCC23)=O)ncc(F)c(-c2ccsc2)n1 37133,C1(NC(C2(CC#C)CC=CCC2)=O)CN(C(c2ccco2)=O)CC1S(C)(=O)=O 37134,c1(SCC(N2CC(C(C)NC(=O)CCOC3CCCCC3)C2)=O)n[nH]c(O)n1 37135,Cn1nc(C(F)(F)F)c(CSC2CC3CC(OC(F)F)C3C2)c1Cl 37136,C(=O)(C1=NOC2(CCN(C(c3ccsn3)=O)C2)C1)N1CCN(C)C(=O)C1 37137,Cn1c(C(=O)NCCCNC(c2c(F)cccc2Br)=O)cc2c1CCOC2 37138,C(=O)(CCCC#CC)NC1CCN(C(C(C)OCC#C)=O)C1 37139,Cc1ccnc(C(=O)NCC2CCN(C(=O)C=C(Cl)Cl)C(C)C2)c1F 37140,c1(CC)ccc(C(N2CCN(C(=O)C=C3CCC3)CC2CC(F)F)=O)c(O)c1 37141,c1(C(=O)NC2CCCC(NC(C3CC(CC4CC4)C3)=O)C2)cccc2ccsc12 37142,CC(CC(=O)NCC1CCCN1C(c1ccc(CO)o1)=O)C(C)(C)C 37143,N1(C(CNC(C(CC)CC)=O)=O)CCCC(NC(c2ccc(F)c(Cl)c2)=O)CC1 37144,C1(C(=O)OC)CC(C(N2CC(OC)C(c3cccc(F)c3)C2)=O)CN(C(C)=O)C1 37145,C1(CC=C)(NC(=O)CC(C)(C)C)CCCN(C(=O)CSc2ccc(C)c(C)c2)C1 37146,CN1C(=O)C2CN(C(c3ncc(CC4CC4)s3)C(=O)NC3CC3)CCN2C1=O 37147,Cn1c(Cl)nc2cc(C(=O)NC3C=CC(C)(C)CC3)ccc12 37148,CCC(C)(C)CC(=O)N1CCCC(C(=O)NC2(C3CCCO3)CC2)C1C 37149,C(C1=NOC2CN(C(=O)C=Cc3cncs3)CC12)NC(=O)COCC1CCC1 37150,Cn1ncc2c(NCc3cnccc3Cl)[nH]c(=NCC34CCCC3C4(F)F)nc12 37151,C#Cc1cn(C)nc1C(N1CC2CC1CN2C(=O)CCCCN1CCCC1)=O 37152,c1(C(N2CC(CNC(=O)C=Cc3cn[nH]c3)C(O)C2)=O)cc(F)cc(F)c1 37153,C(=O)(CCC(N)Cc1ccccc1)N(C(CCC)C)C 37154,C(=O)(CCC(=O)NCC1(O)CC(NC(=O)C=Cc2cccs2)C1)OC(C)(C)C 37155,C1(NC(C2CCC3(CCC3)OC2)=O)CC2CCCC(C1)N2C(C1CSC1)=O 37156,C1(C(N2CC(C#N)(SC)C2)=O)(CC)CCCN1C(C1CCCOCC1)=O 37157,C(=O)(CC(CC)CC)NC(CCCC)CNC(c1ccn(CC#N)n1)=O 37158,c1(CC(=O)NCC(CO)NC(=O)CN2CC3CC3C2)cc(Cl)c2c(c1)OCCCO2 37159,N1(C(c2ccoc2)=O)CC2CC2(NC(C2C(c3ccccc3)C2(F)F)=O)C1 37160,c1(C(C(=O)OC(C)C)NC(=O)NCCc2cn(CC)nc2)ccc(F)cc1 37161,c1(OC)c(Br)ccc(F)c1S(=O)(=O)N1CCC(O)(c2ccccc2Cl)CC1 37162,c1(CC)nc(C)cc(=NCC(CC(C)C)NC(C2CCCCO2)=O)[nH]1 37163,C12(CC(N3C4(CN(CC(c5cnc[nH]5)=O)C4)CC3)=O)CC3CC(CC(C3)C1)C2 37164,c1(C(=O)NC(C2CCN(C(c3cnc(Cl)cc3Cl)=O)C2)C)ccc(C#N)cc1 37165,C1(C(N2CC(c3cc(C)on3)(O)C2)=O)C=CCNC1=O 37166,N1(C(c2cc(OC)ncn2)=O)CCC(CCNC(=O)COCC(F)F)CC1C 37167,c1(N2CCC(NC(N(CC(C(=O)OC)C)C(C)C)=O)C2=O)c(F)cccc1F 37168,C1(CNC(C2CCCC(O)C2)=O)CC2C(C1)C2(F)F 37169,c1(CCSC)nc(-c2nc(Cl)cs2)n(-c2nccn2C)n1 37170,n1(C(CC)C)ncc(C(=O)Nc2nccnc2SC)c1C 37171,C1(CNC(CSCCCC)=O)CC(C(F)(F)F)CN1C(=O)Cc1cncn1C 37172,C1(C(N2C(C(=O)N(C)Cc3cncnc3)(CC)CCC2)=O)C2CC3C(C2=O)C13 37173,CCC(O)C(=O)NC1CC(F)(CNC(c2n[nH]cc2-c2cnn(C)c2)=O)C1 37174,C=CCC(C)(C)C(=O)NCC1CCC(NC(C2CC3CC2C3)=O)CC1 37175,C12(C(=O)NC(CN(C(COCCC)=O)CC)C)CCC(C)(CC1)CC2 37176,C1(NC(c2c(C)onc2)=O)C2CC1N(C(C1(n3cccn3)CCC1)=O)C2 37177,c1(NC)ccccc1C(=O)NC1CC1NC(c1cnc(Br)s1)=O 37178,C#Cc1cncc(C(=O)NCC(C(C)(C)C)NC(=O)Cc2ccsc2Cl)c1 37179,N1(C(c2c(CC)nnc(C)c2)=O)CC2(COC(CNC(=O)C=NOC)C2)C1 37180,C(C)(CC)(CCNC(=O)C(C)Cc1cnn(C)c1)NC(C(C)=C(CC)C)=O 37181,N1(C(C)C(=O)NCC2CC2NC(=O)COC2CCCC2)C(=O)CCC1=O 37182,c1(OC)nc(C)ccc1C(N1CCC(C)C1CNC(C1(C)CC(=O)N(C)C1)=O)=O 37183,C1(C(N(C2CC(SC)C2)C)=O)CCCCN(C(C2CCOC2(C)C)=O)C1 37184,C1(NC(c2cc(CC)no2)=O)CCN(c2ccncc2C(=O)OC)CCC1CO 37185,Cc1sncc1C(=O)N(C(C(=O)NC(c1ccccc1)C)C1CC1)C1CC1 37186,C1(N(CC#C)C(C2CC(C)(C)C2)=O)CCN(C(c2cscc2C#N)=O)CC1 37187,c1(CC(N2CC(C(=O)NCC3CC(=C)C3)(COC)C2)=O)ccc(C)c(F)c1 37188,c1(C(N(CCC)CCNC(=O)C(O)C2CC2)=O)ccc(Br)c([N+](=O)[O-])c1 37189,C1(C(=O)NC(C)C(=O)NC2CCC(N(C)C)C2)OCCCC1(C)C 37190,Cc1cc(NC(=O)NC2CCN(C(N3CCOC3=O)C)C2)cc(C)c1Cl 37191,c1(C(=O)NC2CCCC(CNC(C(CC)(C)C)=O)C2)cc(OC)c(OC)c(N)c1 37192,C1(C(=O)NCC2C=CC(NC(c3n(CC)ccc3)=O)C2)CCc2cnc(C)n2C1 37193,S(=O)(=O)(c1cc(Br)ccc1F)N1CCC(c2ccccc2)(C(=O)OC)C1 37194,Cc1nnc(CCCNC(=O)Nc2csc(-c3ccc(F)cc3)n2)n1C 37195,CC1c2cc(Br)ccc2CCN1CCSc1ccccc1F 37196,c1(C(=O)NCCCN(C(C(SC)SC)=O)C2CCCC2)ccc(C)c(F)c1F 37197,C(C)(C)(C(C)NC(=O)CC(C)c1cnn(C)c1)NC(C(C)C)=O 37198,C1(C(=O)NC2CC(CCC(=O)NCC(C)C#N)C2)CCNC(=O)C1 37199,CN1C(=O)OCC1C(=O)NC1CN(C(c2cn(Cc3ccccc3)cn2)=O)C1 37200,C1(NC(CCNS(C)(=O)=O)=O)CN(C(=O)CC(O)c2ccccc2)C2CCCC12 37201,C1(CC)CN(C)CCN1C(C1(NC(=O)C=Cc2cn(C)nn2)CCSC1)=O 37202,N1(C(CNC(N)=O)=O)CCC(C2(O)CCN(C(C3CCC(=O)O3)=O)C2)CC1 37203,CCC(O)C(=O)N1CCCC1CN(C(=O)Cc1cnc[nH]1)C 37204,CC1(C)CCC(C)(NC(=O)CCNC(c2ccc(F)cn2)=O)C1 37205,c1(NC)nc(C)ccc1C(=O)N(C)CC1CCCC(NC(=O)Cc2ccsc2)C1 37206,CCC(CN(C)C)CC(=O)NC1CN(C(c2cc(C)nc(O)n2)=O)CC12CC2 37207,C12(NC(C(CC)=CC)=O)CC1CN(C(=O)Cc1sc(C3CC3)nc1C)C2 37208,CC1CN2CCN1C(C(=O)NC(C1CCN(C(=O)Cn3cccn3)C1)C)C2 37209,N1(Cc2cc(C)n(-c3cc(OC)c(C)cc3)c2C)CCCC(C2(O)CCC2)C1 37210,Cc1ccnc(C(N2CCC(C(=O)NOC3CCOC3)(C(C)C)CC2)=O)c1N 37211,CCC(C(=O)OC)C(=O)NC1CN(C(=O)Cc2ccc(OC)cn2)C1 37212,c1(CC(=O)NCCN(C(c2ccc(CSC)o2)=O)C2CC2)ccc(F)cc1C 37213,Cc1ccc2snc(C(=O)NCC3CC3CNC(=O)Cc3cnnn3C)c2c1 37214,C(=O)(CN=c1cc[nH]cc1)NC(CC)CNC(=O)C1=C(C)OCC1 37215,N1(C(c2nn(C)c(Br)c2C)C(=O)NCCCSC)CCC2(CNC(=O)C2)C1 37216,N1(C(C(n2c(C)ncc2)C)=O)CCC(C(=O)NCCC2(C)CC2)C1C 37217,C(=O)(C1=C(SC)CCCC1)NCC(CC)NC(c1ccc(Br)o1)=O 37218,N1(C(C(c2ccc(N(C)C)cc2)C)=O)CC(NC(=O)CC2CSC2)CC12CCC2 37219,CC1(C)C2CCC1(CC(=O)NC1(CF)CCN(C(=O)CCC3CCCO3)C1)CC2 37220,C#Cc1ccccc1CC(=O)N(C)CCNC(c1cc(C2CC2)on1)=O 37221,C1(NC(C(C)OCC)=O)CC2(CCN(C(c3cnn(CC)c3Cl)=O)C2)C1 37222,c1(NCC(C)CNC(C2CCCC(C)(C)CC2)=O)cccc(F)c1[N+](=O)[O-] 37223,c1(NC2CC(C)C2)nc2cccnc2c(=NCc2nn(C)cc2Br)[nH]1 37224,N1(C(c2occ(C)c2C)=O)CCCC12CCN(C(=O)CC1CSC1)CC2 37225,C1(C(=O)NCCOCC(N)=O)(CC)CCN(C(=O)C(C)=C2CC2)C1 37226,c1(OC)cc(CC(=O)NC2(C)CN(C(C3CCC(CN(C)C)O3)=O)C2)ccn1 37227,N#Cc1ccc(C(=O)NCC(CC2CC2)C(=O)NCCc2cncs2)o1 37228,C12(C(N(C(CC)CC)CC)=O)CC(NC(=O)C(F)C3CCC3)(C1)C2 37229,N1(c2ccc(C)cn2)CC2C(C1C(=O)NC(=O)CCc1ccccc1N)C2(C)C 37230,C1(C(N2C3C(NC(C(CCC)=CCC)=O)C(C3)C2)=O)CCC([N+](=O)[O-])CC1 37231,c1(C(=O)NC2C3CCN(C(c4c(CC)nc[nH]4)=O)C32)c(Br)ccc(OC)c1C 37232,c1(C(=O)NCCC2OCCN(C(CC=C)=O)C2)cc(OC)ccc1Br 37233,c1(N2CC(C)OCC2)nc(=NCCOc2ccncc2)[nH]c2c1SCC2 37234,C(c1ccc(C)cc1)=CC(N1C(CC)C(C(=O)N(C(C)CN(C)CC)C)CC1)=O 37235,c1(C(=O)NC2CCN(C(C(NC(C)=O)=Cc3cccs3)=O)C2)cc2occc2[nH]1 37236,c1(C(=O)NCC(C)(CC(C)C)NC(COCC(=O)NC)=O)ccnc2[nH]ncc12 37237,c1(CC)cnccc1C(=O)N(CC(O)CNC(c1nccnc1C(F)(F)F)=O)C 37238,c1(C(C)C(=O)N(C)C(c2ccc(Cl)cc2)C2CCCC2)ccc2c(c1)OCO2 37239,C1(C(N(CCC)C(C)C)=O)CC(C(=O)OC)=NO1 37240,C1(NC(C(CC=C)(F)F)=O)CCC2CCN(C(=O)CCCn3cccn3)C1C2 37241,Cc1ncc(CC(N2CCC(NC(=O)C(C)NC=O)C(C)C2)=O)c(O)n1 37242,c1(C(N2CCC(C)(CNC(C3CC(=O)N(O)C3)=O)C2)=O)cc2nc(=O)ccn2[nH]1 37243,N(C1CCCc2ccc(F)cc21)C(=O)NC(C)CCCC(F)(F)F 37244,Cn1cc(I)cc1CN1CC(CN2CCCC2)OCC1 37245,C1(C(=O)NC(CCC)CCO)CCCCN(C(=O)CC2CC(OC)C2)C1 37246,C(=O)(C(C)(O)CC(F)(F)F)N1CC(C)C(n2cc(-c3ccc(CO)nc3)nn2)C1 37247,C(C)(N=c1nc(NCC(C)C(C)(C)C)c2c([nH]1)c(C)nn2C)c1c(C)nc(C)[nH]1 37248,C(=O)(CCC(C)(C)C)NCC1OCCC(NC(CCN2C(C)CCCC2)=O)C1 37249,c1(C(N2CC3C(CNC(Cc4c(C)noc4)=O)(C3)C2)=O)cnc2c(c1)CCCO2 37250,C1(OC)CC(NC(=O)CC(F)F)N(C(=O)CCCC2CN(C(=O)OC(C)(C)C)C2)C1 37251,CCC(CC(C)C)C(=O)N(CC(O)CNC(c1ccc(Br)c(Cl)c1)=O)C 37252,c1(C(C(=O)NCC2C(OC)CCC2)(C)C)ccc(C(F)(F)F)cn1 37253,C12(C(=O)NCC3(N(C)C)CCCC3)CC1CCN2C(c1cnc[nH]c1=N)=O 37254,c1(C(=O)NCC2C(NC(CC3(C)CCCO3)=O)CC2)nccc(Cl)c1F 37255,N(C1CCCc2n[nH]cc21)C(C(CO)NC(CCC(C)(F)F)=O)=O 37256,CCCCC(CCCC)C(=O)N1CC(NC(=O)C(C)(C)NC(=O)C(F)(F)F)C(C)C1 37257,C=CCN=c1nc(N2CCOC(CNC(=O)C(C)C)C2)c2ccc(OC)cc2[nH]1 37258,Cc1c(C(=O)NCCCCCCNC(=O)CN2CCCC2=O)c(C(F)F)nn1C 37259,N1(C(c2cn(C(C)C)nn2)=O)CCC(C)(C)C1CC(=O)NC(C(F)(F)F)C1CC1 37260,C1(CNC(C=CC=CC)=O)C2CN(C(C3CCCN3c3ncccn3)=O)CC12 37261,c1(OC)cccc2[nH]cc(CC(N3CCCC(C)(C(=O)NC4CC4C)C3)=O)c12 37262,c1(NC)ncccc1C(N1CCC(F)(C(N2CCC(CN(C)C)C2)=O)C1)=O 37263,C#CC1CN(C(C2CC3(C2)CC(O)C3)=O)CCN1C(c1cc(C2CC2)on1)=O 37264,C1(NC(=O)CC2CCCCC2)CC1C1CCN(C(c2nnc(O)cc2O)=O)CC1 37265,C1(C(N(C2CCC(O)C2)C)=O)CCOC2(CCN(C(=O)OC(C)(C)C)CC2)C1 37266,CC1CN(C(C(=O)NCc2ccco2)c2cnsc2)CC(C2CC2)O1 37267,CCC(N=c1nc(N2CC3CC2CN3C)c2[nH]ccc2[nH]1)c1ncc(C)[nH]1 37268,N#Cc1ccc(CN2CCC(O)(C(=O)Nc3cc(Cl)ccc3I)C2)cn1 37269,N1(C(c2nnn(CC)c2C)=O)CC2CCC1C1CN(C(=O)CC(F)(F)F)CC21 37270,c1(C(=O)NC2C(CNC(=O)CC3CCC(C4CC4)O3)CC2)ccc2c(c1)OCC2 37271,N1(C(CC2C(C)(C)C2(C)C)=O)CC=C(CC(=O)NC2C=CCCC2CO)CC1 37272,c1(CSC)cccnc1C(=O)NC(C)CC1CN(C(C2COCCOC2)=O)C1 37273,C(=O)(C(C)(C)CCCC(=O)NCCCNC(=O)CCC1CC(C)(C)CO1)OC 37274,C(=O)(C1=CCCCO1)N(C1CCCN(C(C(=CC2CCCC2)C)=O)C1)CC1CC1 37275,C1(C(=O)NC2(C)CC(NC(C3C(CCC)C3)=O)C2)CCC(O)(c2ccccc2)C1 37276,CC1(C)CC(O)(C(=O)NCC2CCCN(C(c3ccc(CO)s3)=O)C2)C1 37277,Cc1cccc([N+](=O)[O-])c1N1CCCC(C)(CNC(C2(CF)CCC2)=O)C1 37278,c1(C(=O)NCC(CO)NC(c2sccc2F)=O)cccn2nncc12 37279,N1(C(=O)CC2CCOCC2)CCCCC(C2CN(C(C3CCSC3)=O)C2)C1 37280,C1(OC)CC2CC1CC2C(=O)Oc1snc2c1CCC2 37281,N1(C(c2c(C(C)C)onc2)=O)CC2CCC2(CNC(C2CCS(=O)(=O)CC2)=O)C1 37282,N1(C(c2ccc(SC)cc2)=O)CC=C(CNC(=O)C(C2CCOCC2)O)CC1 37283,CCCCCC(=O)NC1CCOC(CNC(=O)C(O)c2cnc[nH]2)C1 37284,CC(CNC(c1cc(CCO)on1)=O)C(F)C(=O)NC1CCC(O)C(O)C1 37285,C1(CCNC(C2C(OC)CCC2)=O)C(C)CCCN1C(=O)C1=CCN(C)C1 37286,C1(C(N2CC(F)(CNC(C3C(C)CC3)=O)C2)=O)CC2C=CC1C21CC1 37287,C1(CNC(CC(=C)C)=O)(OC)CCS(=O)(=O)CC1 37288,C1(CC(C)(C)C)CN(C(c2scnc2C(F)F)=O)CC1NC(=O)C=CCF 37289,N1(C(CC(CC)(F)F)=O)CC(C2CCCCN(C(C3C4(CC4)C34CC4)=O)C2)C1 37290,C(=O)(CC1=NN(C)C(=O)C1)NCCN(C1CCCCC1)C(C1C(C)SCCC1)=O 37291,C#Cc1ccc(Cl)c(C(N2CC(NC(=O)C(F)F)C(CC)C2)=O)c1 37292,N1(C(CC(C)(C)NC(C2C(C(C)=O)C2(C)C)=O)=O)CCCC2CC1C2(C)C 37293,CCCCCCn1nnnc1C(CCC1CCCCC1)NC(CC)CCC 37294,Oc1c(F)ccc(CN=c2ccnc(N3CCC(c4ccncc4)CC3)[nH]2)c1F 37295,Cn1nc2ccccc2c1C(N1CCCN(C(=O)Cn2cnnc2)C(CO)C1)=O 37296,N1(C(CC2N(C)CC=CC2)=O)CCC2CN(C(c3ncccc3Cl)=O)CC2CC1 37297,C1(NC(C(CC)OCC)=O)C2CCN(C(C3CC(C4CCC4)C3)=O)CC12 37298,C1(CNC(c2cc(CC)nn2C)=O)CC2(CCN(C(=O)C=CC3CC3)C2)CO1 37299,c1(CNC2C(C(=O)OC)COCC2)nc2ccccc2n1CC(F)F 37300,C1(CNC(C(C)Cc2ccc(C#N)cc2)=O)CCC(C)(C)CN1CC1CCCO1 37301,CCCCC(C)C(=O)NCc1n[nH]cc1C(=O)Nc1cscc1CC 37302,c1(C(=O)OC)cc(C(=O)NCC(C)CNC(c2ccc(F)s2)=O)c(F)c(F)c1 37303,N1(C(C(=O)NCC)=O)CCC2CN(C(c3ncnc(OC)c3F)=O)CCC2C1 37304,C12(CNC(c3n(C(C)C)cnc3)=O)CC(CO1)N(C(C1CCN(C)C(=O)C1)=O)C2 37305,Cc1nn(C)c2ncc(C(N3CCC4(NC(c5cccnn5)=O)CC4C3)=O)cc12 37306,N1(C(C2C(C)=CCS2)=O)CCCC(C(N2CC(O)(c3cnn[nH]3)C2)=O)C1 37307,C(=O)(CC(C)CCC(=O)NCC(CC(C)C)NC(c1cnn(CCF)c1)=O)OC 37308,C(=O)(CCCC(C)(F)F)NCCN(C(=O)CCOCC1CCCO1)C(C)C 37309,CC1(C)CC(NC(=O)CCOC2CCOCC2)CN(C(c2ccncc2O)=O)C1 37310,C(c1cccc([N+](=O)[O-])c1)=CC(=O)NC(CN(C(=O)C(C)(C)C(F)(F)F)C)(C)C 37311,Cc1nc(CO)ncc1C(=O)NC(CNC(=O)CC1CC(F)(F)C1)C(C)C 37312,C12(C(=O)NC(COC)C(=O)OC)CC(C)(CN1C(=O)C(F)C(F)(F)F)C2 37313,c1(C(N2C(C)CC(CNC(c3cc(Cl)c(Cl)s3)=O)C2)=O)cc2ccccc2cn1 37314,N1(C(CC(CC)C)C)CCCOC(NC(C)(C)Cc2ccccc2)C1.C1C(=O)N1 37315,C1(CC(=O)NCC(CC(=O)OC)O)CN(C(c2ccccc2O)=O)CC12CC2 37316,c1(C(N2CC3N(C(C4N(CC)CCOC4)=O)C(CC3)C2)=O)c[nH]c2nccc-2c1 37317,C1(C(=O)NC(CC)CN(C)C(c2sccc2CO)=O)CCn2cnnc2C1 37318,CC(C)C(CO)C(=O)N1CCC(NC(=O)Cn2nnc(C3CC3)n2)C1C 37319,C(=O)(C(C)CC(C)C)N1C(CCC(=O)NC(CC#C)CC#C)CCC1 37320,C1(C(=O)NC(C2CCCOC2)C)CCCC(NC(C2(NC(N)=O)CCC2)=O)C1 37321,C(=O)(C(O)CC(F)(F)F)NCCCN(C(C1(C)CC(F)(F)C1)=O)CC 37322,c1(C(=O)NC(c2cn(CC)nc2)C)cncnc1C1CC1 37323,Cc1nc(C(N2CCCC2CCSC2CCCC2)C(=O)NCC2CC2)oc1C 37324,C1(NC(=O)C=CC2CCCC2)CC2CCC1(NC(C1(F)CCCCC1)=O)C2 37325,c1(C(N(CCOCCN(C(C(=O)NCC)C)C)C)=O)nccc(C)c1N 37326,C1(NC(C=CSC)=O)CC2(C1)CC(CNC(c1cc(C3CC3)nc(O)c1)=O)C2 37327,C1(CC(=O)NCC2(C)CC(NC(=O)CN3CC4CC4C3)C2)CCCCC1(F)F 37328,C1(CNC(C(=O)NCC(F)F)=O)CC2COCC2N1C(c1ccc(C(F)F)[nH]1)=O 37329,C1(C(N2C(C)(C(=O)OC)CC2)=O)CCN(C(C2C3CCCC23)=O)CC1(C)C 37330,C1(C)(C(=O)NC(C)Cc2ccco2)CCCCC1(C)C 37331,C(CC(O)C(=O)NCC(C1CCC1)NC(c1ccc(-n2ccnc2)nc1)=O)SC 37332,C1(CC(=O)NCCN(C(c2cnsc2)=O)CC)CC(C)(C)CCO1 37333,c1(C(N(CCCOCCNC(C2COCCO2)=O)C)=O)ccc2nn(C)cc2c1 37334,c1(C(=O)Nc2ccnc3ncnn23)cc(-c2ccccc2)nc2ccccc12 37335,C1(C(N2CC(CNC(CP(C)(C)=O)=O)OCCC2)=O)CCOCC12CCCCC2 37336,C1(C)(C(N2CCOCC(NC(CCC=CC)=O)C2)=O)CC2CCC(C1)S2 37337,N1(C(c2ccc(Cl)cc2F)C(=O)NC(CC)(C)C)CC(C)OCC1(C)C 37338,N1(C(C2=CCCCC2C)=O)CCn2nc(CNC(c3cccs3)=O)cc2C1 37339,C1(O)(C(C)NC(=O)Cc2ccn(C(F)F)n2)CCN(C(C2CNC(=O)N2C)=O)C1 37340,c1(C(N(CC(C)NC(c2ccnc(C(C)(C)C)c2)=O)C)=O)cncc(Cl)c1Cl 37341,c1(CCC(=O)NCC(CNC(=O)C(C2CCCCC2)O)OC)ccc(C#N)cc1 37342,c1(C(CNC(COCCC=C)=O)NC(=O)CC2(C)CCOC2)cc(F)cc(Cl)c1 37343,C1(NC(c2ccon2)=O)CCCOC1C1CCN(C(=O)CN2CCCC2=O)CC1 37344,N1(C(C(C(=O)OCC)F)=O)CCC(C)(CNC(c2ncn(C(C)(C)C)n2)=O)CC1 37345,N1(C(C=CC=CC)=O)CCCC(CO)(NC(=O)C(C)C2CCOC2)C1 37346,c1(C(C)SCC)nc(-c2oc(CC)nc2C)n(-c2ccn(C)n2)n1 37347,CC1CN(C(c2cccc(C(C)(C)C)n2)=O)CCN1Cc1cc(Cl)ccc1F 37348,C1(C)(C(=O)NC(CC)C(F)(F)F)CC(O)CN1C(c1ccc(=N)[nH]c1)=O 37349,N1(C(c2cc3cscc3s2)=O)CCC(C2CCCN(c3ncncc3I)C2)CC1 37350,c1(C(=O)NC(C(=O)N2CCC(CC#C)C2)(C)CSC)cc(C)ncc1C 37351,N12CCN(C3CCC13)C(=O)CSCC(C)C2=O.c1(CSC)nccn1C(C)(C)C 37352,C1(C(N(CC(C2CC2)OC)C)=O)CCN(C(c2nc[nH]n2)=O)C1C 37353,Cc1ccc(F)c(C(N2CCC(O)CC2C(=O)Nc2ccccc2)=O)c1Cl 37354,c1(C(=O)NC2CCCC2)occ2c1CCC2.Cc1cc(C(=O)N2CCC2)ccn1 37355,CC1CN(C(C2(C(C)(C)O)CC2)=O)CCC1C(=O)NCCC1CCC(C)(C)C1 37356,C1(C(N2CCC(CC(N3CCN(C(C)=O)CC3)=O)CC2)=O)CCC2(CCC2)C1 37357,C1(F)(C(=O)NCc2ccc(C(N)=O)s2)CCCN(C(C2C3COCC23)=O)C1 37358,c1(C2(C(=O)NCCC3CN(C(C(C)NC(C)=O)=O)C3)CCC2)ccccc1F 37359,C1(CNC(C(C)OCC(C)C)=O)C2CCCC1N(C(C1CCCS1)=O)C2 37360,C1(NC(C2(C)COC2)=O)CC(F)(F)CC1NC(c1ccc(CN2CCCC2)o1)=O 37361,Cc1ccccc1-n1ccc(COC(c2ccc(C(F)F)nc2)=O)n1 37362,CCCCCCC(C)(CC)c1nc(Cc2ccc(C)nc2)no1 37363,N1(C(C2(OC)CC2)=O)CCC(c2cc(CNC(C34COCC3C4)=O)on2)CC1 37364,c1(CCC)cnnc(C(=O)NC2CN(C(c3cc[nH]c3C3CC3)=O)CC2OC)c1 37365,c1(OC)cnncc1C(=O)NCC(O)CNC(C1(O)CCCCC1)=O 37366,C1(NC(=O)Cc2cscn2)CN(C(c2csc(O)n2)=O)C2(CCCCCC2)C1 37367,C(C(=O)NCC(CC)NC(C1C(=C)C1)=O)(C(C)OC)NC(=O)OC(C)(C)C 37368,C1(CNC(c2cc(CC)nn2C)=O)CCCC2(CN(C(=O)C3=CCSC3)C2)O1 37369,Cc1cc(C(=O)NC2CCCC2CNC(c2cccnn2)=O)c2c(c1)CCO2 37370,[N-]=[N+]=NC1CCC(NC(=O)NCC2CCN(C(=O)CCCCN3CCCC3)C2)C1 37371,c1(N(C(CNC(c2c(C)nn(CC)c2C)=O)C)C)nc[n+]([O-])cc1[N+](=O)[O-] 37372,CCCCCC(=O)N1CCC(C(=O)N(CCCCN(C)C)C)C1C 37373,C1(CNC(C(c2ccc(C)s2)C)=O)CC(F)(F)CN1C(C1CN2CCN1CC2)=O 37374,c1(SC)ccc(C(=O)NC2(CNC(=O)C#CC3CC3)CCCCC2)cc1 37375,CCCCCC(O)C(=O)N1CC2CC1(CNC(C1CC1CN(C)C)=O)C2 37376,c1(C(C2(CC)CC2)(C)C)nc(-c2cnn(C)c2)nn1CC1CCCC1 37377,CCN=C(NCCc1ccsc1Br)NCC(c1ccoc1)O 37378,c1(C(=O)NCCN(C(=O)CC2(O)CCC2)CCOC)scc(C)c1C 37379,C(C)(CC(C)N=c1cc[nH]cc1C#N)NC(c1c(O)nnc(CC)c1CC)=O 37380,CC#CCCC(=O)NC1CCCC(NC(=O)CCOc2ccc(Br)cc2)C1 37381,c1(C(=O)NC2(CC=C)CCN(C(=O)C(CCO)NC)C2)oc2ccccc2c1C 37382,N1(C(CCCC#C)=O)C2CCCC1CC(CNC(c1ccccc1C)=O)C2 37383,c1(CCC(=O)NC2CN(C(C3(OC)CCSC3)=O)C(C)C2)c(C)nn(C)c1C 37384,C1(NC(C23COC(CF)(C2)C3)=O)CCN(c2cnccn2)CC1 37385,c1(C(N2CCCN(C(C3(C)ON=C(C)C3)=O)CC2)=O)cc2c(s1)C(C)(C)CCC2 37386,N1(C(C2=C(C)OCC2)=O)CC(NC(=O)C(C)CS(C)(=O)=O)C2(CCOCC2)C1 37387,C1(CNC(c2ccco2)=O)CC2CCCC2N1C(C1C(F)(F)C12CCC2)=O 37388,c1(CCS(=O)(=O)N2CCCC2Cc2cccnc2)ccc(F)c(Cl)c1 37389,C1(C2CCCN(C(c3cc4ccc(F)cc4s3)=O)C2)(NC(CC2C(C)C2)=O)CC1 37390,O=C(C1=CC2(CCOC2)C1)N1CCC(F)C(NC(C2(C(F)(F)F)CC2)=O)C1 37391,N1(CC(N2C(C3(NC(CCCC)=O)CC3)CCC2)=O)CCCNC1=O 37392,N1(S(CCC)(=O)=O)CCN(C(C2CC2(F)F)=O)CC12CC2 37393,c1(CCC(=O)NC2(C)CN(C(c3cc4n(n3)CCC4)=O)C2)cccc(Cl)c1Cl 37394,N1(C(C(C)NC(=O)C(F)(F)F)=O)CCC2CN(C(c3ccccc3C#N)=O)CC12 37395,c1(C(=O)NCC2CN(C(Cc3scc(C)c3)=O)C2)cccc2cccnc12 37396,C1(CNC(=O)NC(c2onc(C)n2)C(C)C)CC2(CC2)C(=O)O1 37397,Cc1nc2c([nH]1)CN(C(C1CCCN1C(C1CC1Cl)=O)=O)CC2 37398,C1(C(=O)NCC=CCNC(C2C(OCC)C2)=O)CCC(C2CCC2)CC1 37399,C1(C(=O)NC2(C(N)=O)CCC2)C=CCN1C(c1cccs1)=O 37400,c1(CC)cc(F)ccc1C(=O)NC1CC(NC(c2nc(C)ncc2Cl)=O)C1 37401,S(=O)(=O)(c1ccc(Cl)nc1)N1CC2(CC(C(=O)NCCc3c(C)ncs3)C2)C1 37402,C1(C(F)(F)F)(NC(C(N2C(CNC(C(N)=O)=O)CC2)=O)=O)CC2(CC2)C1 37403,C1(NC(CCn2ncc(C)c2)=O)CC2CC1N(C(=O)CCNC(=O)CO)C2 37404,Cc1cc(=O)oc2cc(N(C(C)C(=O)N(C)CCN3CCCC3)C)ccc12 37405,c1(-c2ccc(NC(C34CNCC3C4)=O)s2)cccc2ccccc12 37406,c1(C(=O)NCCN(C(C2(C(=O)OC)C=CCC2)=O)C)cc2c(cc1Cl)NC(=O)C2 37407,c1(CNC(c2cc(F)ncc2F)c2n(CCSC)nnn2)nc2ccccc2s1 37408,N1(C(C(CC=C)C(=C)C)=O)CCC2(CCC2NC(=O)C(C)(C)C(C)=O)CC1 37409,N1(C(C(CO)N(C)C)=O)CCCC(C2CCCN2)C1.c1(C(C(C)CCl)=O)cc(Cl)n[nH]1 37410,Cc1cc(F)c(O)c(CN2CCCC2c2nnc(O)o2)c1 37411,N1(C(=O)CCc2ncccn2)CCN(C(=O)CC2CCCC2(F)F)CC1 37412,C12(C(=O)NC3CC(C)(CNC(C=CC)=O)C3)CCCCC(=O)N1CCC2 37413,S(=O)(=O)(c1cncc(Br)c1)NCC1(C)CN(Cc2cc(F)ccc2Br)C1 37414,c1(C(N2C(C(=O)Nc3c(C)cccn3)CCC2)=O)ccc([N+](=O)[O-])c(N(C)C)c1 37415,Cc1ccc(C(=O)N(C)CCNC(C2CCOC2=O)=O)cc1OC(F)F 37416,C12(CC)CCCN1C(=O)CC(=O)NC2=O.N1(C(C)=O)CCCC1.OC 37417,c1(N(C)C(C2CC(NC(=O)OC(C)(C)C)C2CC(=O)O)=O)cnccc1Br 37418,c1(C(N2CC3C(NC(C4CC5OCCC5O4)=O)C3C2)=O)cccc2ccoc12 37419,Cn1c(CC(=O)NCC(C2CC2)NC(=O)CC2(C(F)(F)F)CC2)nnc1S 37420,C(=O)(C(CCC1CCC1)NC(N)=O)N1CC(CCC(C)NC(=O)C(C)C2CC2)C1 37421,N1(C(C2CC(n3cc(COC)nn3)C2)=O)CC(CN(C(C)(C)C)C)OC(C)(C)C1 37422,N1(C(C(F)=CC)=O)CCCOC(CNC(=O)CC2COC(C)(C)CO2)C1 37423,c1(C(=O)NCC(CO)NC(=O)CC2COCCO2)ccc(-c2nnc(S)o2)cc1 37424,C1(C(N2CCC(CN(C(COC(C)=O)=O)C)CC2)=O)CCC(C)=C(C)C1 37425,c1(C(=O)NCC(CNC(C2C(C)=CCS2)=O)(C)F)cc(N)c(O)c(F)c1 37426,c1(OC)ccc2ccccc2c1C(=O)Nc1csc(-c2cc(SC)ccc2O)n1 37427,C(CCCC(=O)NCC1(CC)CC(NC(=O)CCc2ccncc2)C1)OCC 37428,CC(C)CC(CNC(=O)CC1CCCCO1)NC(C1CC(O)CN1C(N)=O)=O 37429,C(CCCCCC(=O)NOCC1CCC1)NC(Cn1c(C)nnn1)=O 37430,O=C1CC(C(N2CCC(OCCF)C2)=O)N(C(=O)C(=C2CCCCC2)F)C1 37431,N1(C(C(n2cc(CCCSC)nn2)C)=O)CC(C(N)=O)C(c2cnn(C)c2C)C1 37432,N1(C(c2ccc(C(N)=O)cn2)=O)CC2(CCN(C(=O)CN3CCCCC3)C2)C1 37433,c1(CN(C2CC2)CC2(C)CCCC2)cncc(C(F)(F)F)c1 37434,C1(NCC2CC(C)(C)CC(C)(C)C2)CCOC2(CCCCC2)C1 37435,c1(N(C2CCN(C(=O)OC(C)(C)C)C2)C(C2N=C(C)SC2)=O)cc(C#N)ccc1C 37436,c1(CC(N2C(C)C(NC(c3cnc(O)n3C)=O)CC2)=O)cc(F)cc(F)c1 37437,Cc1cc(F)cc(Br)c1C(=O)NCC1(c2ccccc2)CCN(C)C1 37438,C(=O)(C(CCOC)OC)NC(C1(CNC(CCOCC#C)=O)CC1)C 37439,N1(C(=O)Cc2cccc(Cl)c2)CC2(CCC(NCc3cnccc3Cl)C2)C1 37440,N1(C(c2cc3ccoc3s2)=O)CC2CCN(C(=O)CN3CCCC3)CC2C1 37441,C1(CCNC(C)(C)C)C2CC3CN(C(=O)NC4(CO)CCC(C)CC4)C1C3C2 37442,c1(OC)ccc(CCNCC(O)C(C)c2ccccc2)c(F)c1F 37443,C(=O)(C1=CCCC1(C)C)N1CCC(O)(CNC(CC2CCN(OC)CC2)=O)C1 37444,C1(CNC(C2(CC#C)CCC2)=O)C(O)C(O)CN1C(=O)CSCCOC 37445,C1(C)(C(=O)NC(C(C)NC(C2CCSCC2)=O)CO)Cc2ccccc2NC1=O 37446,c1(OC)ccc2c(c1)CC(C(N1CC3C(CNC(=O)CC(C)C)C3C1)=O)CO2 37447,c1(CC)ccc(F)c(C(=O)NCC2CCCC(NC(=O)CC3CCOCC3)C2)c1 37448,CC(C)CC(O)C(=O)NCCN(C(=O)CCc1nc(-c2ccco2)no1)C 37449,N1(C(CCCCSC)=O)CCCC(C2CCN(C(=O)C3CC3)CC2)CCC1 37450,Cc1nc(C(N2CC(NC(c3ccnc(O)c3)=O)CC(F)C2)=O)c(C)n1C 37451,N1(C(c2c(Cl)ccc(C)c2)=O)CCC(C2CC2)C1CNC(=O)C(N)=O 37452,C1(NC(C2CC(CNC(CC3(CC(=O)OC)CC3)=O)C2)=O)NC(=O)OC1(C)C 37453,N1(C(Cc2cc(C)on2)=O)CCC(C(=O)NCC2CC(C)CO2)C(C)(C)C1 37454,C1(CNC(C(CC)OCC)=O)(OC)CCN(C(C2CCC3(CC2)N=N3)=O)CC1 37455,C1(CC(=O)OC(C)C(=O)NC(c2ccc(Br)cc2)C)CCCCCC1 37456,C1(NC(c2cncc(-c3ccc(Cl)cc3)c2)=O)CCC(O)(c2ccccc2)CC1 37457,N(C1CCc2cc(Br)ccc21)(C(c1cc(C)cc2cccnc12)=O)CC 37458,CCCCCCCN=c1nc(N2CCC(C(N)=O)(N(C)C)C2)c2c([nH]1)COC2 37459,C12(NC(=O)Nc3cc(CN4CCOCC4)cc(F)c3)CCC(O)(CC1)CC2 37460,N1(C(CN(C(COC)=O)C)=O)CC=CC(NC(C2CC3CCC2C3)=O)C1 37461,Cc1cc(C(N2CC(O)(CCNC(=O)CCS(C)=O)C2)=O)c(C)s1 37462,N1(C(c2cc(C)nc(O)c2)=O)C2CCC1CC(CNC(c1cn(C)nc1Cl)=O)C2 37463,N(C(=NCCCCl)N1CCC2(CNC(=O)C2)C1)CC(C)(O)c1cccs1 37464,c1(Cn2cc(COCC)nn2)cccc(C(=O)N(CC(C)(C)COC)C)c1 37465,C1(OC)CN(C(c2cn(C)nc2Cl)=O)CC1NC(c1ccccc1O)=O 37466,C1(N(C(C(c2cnn(C)c2)OC)=O)C)CCC2CN(C(=O)CCC(C)(C)C)CC12 37467,CC1CN(C(c2cccc(C#N)n2)=O)CCN1C(=O)CCOC1CCCCC1 37468,Cc1ccc(C(C)NC(=O)C(=O)NCCC2COCC2(C)C)cc1C 37469,N1(C(C(C2CCOCC2)C)=O)CCC(NC(=O)C(C2CC(C(=O)O)C2)C)C(C)(C)C1 37470,Cc1ccc(O)c(C(N2CC=CC(NC(c3cc(=O)cc[nH]3)=O)C2)=O)n1 37471,N1(C(C(=Cc2cccs2)C)=O)CCCOC(CCNC(c2csc(O)n2)=O)C1 37472,Cc1sc(C(=O)NC2CCCC(NC(=O)CC(C)NC(N)=O)C2)nc1O 37473,c1(OC)c(C(=O)NC(C2CCCN2C(c2ncccc2O)=O)C)c(C)nn1C 37474,c1(C(N2CC(OC)(CNC(C3(NC(C)=O)CC3)=O)C2)=O)cn2ccnc2s1 37475,Cc1cc(C(N2CC=C(CCNC(=O)CC(O)C3CC3)CC2)=O)c2n[nH]cc2c1 37476,C1(CCNC(C(C(=C)Cl)(C)C)=O)CCN(C(c2ccc(F)cc2O)=O)CC1(F)F 37477,C(N=c1cc(Cl)nc[nH]1)c1c(NC(=O)C(N2CCCCCC2=O)C2CC2)cccc1 37478,CCCCC(O)C(=O)N1CCCC(NC(c2ccc(C(=O)OC)cn2)=O)CC1 37479,N1(C(C(c2ccc(C)o2)C)=O)CCC(C)N(C(=O)COc2cn[nH]c2)CC1 37480,C1(CCC(=O)NC(CN(C(C=CCN(CC)CC)=O)CC)C)CCOCC1 37481,C=CCC(CC)C(=O)N1CCC(n2cccn2)(C(=O)Nc2csc(C#N)c2)CC1 37482,CCC(C)C=CC(=O)N(CC(=O)N(C1CCC1)CC1CCC1)CC 37483,c1(NC(C)=O)c[nH]c(C)c1C(=O)NC1CC(CCNC(=O)CC2CC(F)(F)C2)C1 37484,Cc1ccc2[nH]cc(CCNC(C3C=CCN3C(c3cc(CO)on3)=O)=O)c2c1 37485,c1(OCC)ccc2ccccc2c1NC(=O)C(=O)NC1CCc2nc(C)nn2C1 37486,CCCCC(COC)(c1nnnn1C1COC1)NCc1cncc(C)c1 37487,N1(C(=O)OC(C)(C)C)CCCC1C(=O)NC1CCCC1NC(C1(C)CC=CC1)=O 37488,C1(NC(=O)CCc2ccon2)COCC1NC(c1n[nH]cc1Cl)=O 37489,CC(C)C1=NOC(C)(C(N2CCC(C)(CNC(=O)C=C(C3CC3)C3CC3)C2)=O)C1 37490,N1(C(c2cncc(C)c2)=O)CC(NC(=O)Cn2ncn(C)c2=O)C(F)(F)C1 37491,c1(C(C(N2CCC(CO)(NC(C3CC(O)C3)=O)CC2)=O)O)cccc([N+](=O)[O-])c1 37492,C(C)(N=c1[nH]c(=NCc2nnn(C)n2)[nH]c2c1CCCCCC2)c1c(C)ncs1 37493,C1(NC(COc2ccn(C)n2)=O)CC(F)CN(C(=O)Cn2cnc(=N)[nH]2)C1 37494,N1(C(CC2(CC(=O)OC)CC2)=O)CCCC(NC(=O)Cc2cccc(C)c2)CC1 37495,C(C(C(=O)NCCC1CC(=O)N(C)C1)C(C)(C)C)NC(c1cn(CC)nn1)=O 37496,CN1CCN(C(C2(F)CCCN(C(c3cc(N)cc(F)c3)=O)C2)=O)C(C2CC2)C1 37497,c1(-c2occ(CC(N3CC(CNC(C(C4CC4)OC)=O)C3)=O)n2)ccc(Cl)cc1 37498,C1(C(N(C2CCN(c3ncncc3C)C2)CCC)=O)CC(C)(C)CC(C)(C)C1 37499,C(=O)(CCCc1cncs1)NCC(CC)NC(=O)CSc1nc[nH]n1 37500,C1(C)(CNC(CC(C)O)=O)CN(C(=O)C(=O)C(C)(C)C)CCO1 37501,c1(C(=O)NCC(C)NC(c2cnoc2C2CC2)=O)cnc2c(c1)CCC(=O)N2 37502,C1(NC(N)=O)CC(C(F)(F)F)CN1C(=O)CCNC(=O)Oc1ccccc1 37503,c1(-c2cc(C(N3CC(NC(C(CC)F)=O)C3)=O)on2)c(F)cccc1F 37504,Cc1nccc(=NCC2CCC(CNC(C3CCC(N=[N+]=[N-])C3)=O)CC2)[nH]1 37505,N1(C(c2c(OC)ccc(C)n2)=O)CC(C)(CNC(C2CCCCS2)=O)CC1(C)C 37506,Cc1noc(C)c1S(=O)(=O)N(C1CCCN(C(C2CCCCC2)=O)C1)CCO 37507,Cc1sc(C(F)(F)F)nc1C(=O)N(CC(C)(C)NC(=O)CC1C=NN(C)C1=O)C 37508,c1(C(=O)NC2(C(=O)NC(c3ccnc(C)n3)C)CSC2)cc(O)nc(C)n1 37509,c1(CNC(C(c2sc(Cl)cc2Cl)N(CCC(=O)OC)C)=O)ccccc1Br 37510,CC(C(=O)N1C2CC(F)C(C2)C1C(N1CCCC(F)C1)=O)S(=O)c1ccccc1 37511,C(C(C(C)(C)C)NC(=O)C(O)C1CC1)NC(C=C(C)C(F)F)=O 37512,c1(CNC(=O)NC2C(CCC)C2)cccnc1 37513,CCS(=O)(=O)CC(=O)NC(C)(CNC(=O)C(c1c(C)nn(C)c1C)C)C1CC1 37514,CC1(CC(N2CCOC(CNC(=O)CNC(N3CCCC3)=O)C2)=O)CCS(=O)(=O)N1 37515,O=C(C1CCc2nccn21)NCCC1CN(C(c2ncc3c(F)cccn23)=O)C1 37516,c1(OC)ccc(CN2CCN(C(N)=O)CC2)c(Br)c1O 37517,c1(COCC(=O)NCc2cccc(CNC(=O)C3=CCC3)c2)cc(F)cc(F)c1 37518,c1(N2CCC(CNC(C(c3cccnc3)C)=O)C2(C)C)ccc([N+](=O)[O-])cn1 37519,C(=O)(CCCCCS(N)(=O)=O)NC1CCCCN(C(c2c[nH]c(=N)s2)=O)C1 37520,c1(OC(C(CC)C)C)cc(C#N)ccc1OC(=O)OC(C)(C)C 37521,CCCC(C(=O)NCC1(O)CCCN(C(=O)C2=NOCC2)CC1)S(N)(=O)=O 37522,C(C(C)(C(=O)N(C1(C(N2CCSC(C)C2)=O)CC1)C)OC)OC 37523,c1(C(c2n(CCSC)nnn2)NCC2CCCS2)ncccc1C 37524,c1(CC(=O)NCC2C(NC(C(C)OCCC=C)=O)CCC2)cn2ccccc2n1 37525,c1(NC(=O)NC(c2ccc(C(C)C)cc2)C(C)C)nc2c(O)ncnc2s1 37526,c1(C(N2CC(NC(c3coc(Cl)n3)=O)C(O)C2)=O)nc2ccccc2o1 37527,N1(C(c2c(OC)cncn2)=O)CCC2(CC1)CN(C(=O)CC(C)(C)F)C2 37528,N1(C(CC(C)SC)=O)CCOCC(CNC(=O)CN(c2ncccn2)C)C1 37529,N1(C(CCC(C)=O)=O)CCC(O)C(C(=O)Nc2cc(C(F)(F)F)cc(F)c2)C1 37530,N1(C(C(CC)(C)OC)=O)C2CCC1CC(NC(C13CCC(N=[N+]=[N-])C1C3)=O)C2 37531,c1(NC(C)C)nccc(=NC2CC2C(N2CCC(OC3CCCCC3)CC2)=O)[nH]1 37532,Cc1c(F)ccc(N)c1C(=O)NCC12CC(NC(=O)COC(F)(F)F)(C1)C(C)O2 37533,C=Cn1nccc1C(=O)NC1CC(C)(NC(C2CCCN(C(=O)OC)C2)=O)C1 37534,C(C(=O)N=S(C)(=O)c1cnn2c1CN(c1ncnc(C(C)(C)C)n1)CC2)=CC 37535,c1(C(=O)NC)cc(C)[nH]c(=NCC2CCC(NC(=O)C(C)(C)CC(F)(F)F)C2)n1 37536,N1(C(c2c(C)ncnc2)=O)CCOCC(C)(CNC(=O)Cc2cnoc2)C1 37537,CN=S(C)(=O)c1ccc(C(=O)NCC2CCCCC2NC(c2cccs2)=O)cc1 37538,CC1CN(C(C2CSCN2C(C2(F)CCCCCC2)=O)=O)CC2(CCC2)O1 37539,Cc1cnc(F)cc1C(N1CC(NC(=O)Cc2conc2C)C(C)C1)=O 37540,N1(C(C(N2CC(C)C2)C)=O)CCC(C)(C)C(C(=O)NC2CC(C)(C)OC2=O)C1 37541,C12CC3C(C3C1)NC(=O)CN(C)CC(=O)N2.CCCCCOCC(=O)NC(C)C 37542,CC1=NOC(C)(C(=O)NCC2CCCC2NC(=O)COC(C)(C)C(F)(F)F)C1 37543,c1(CC)c(C(=O)N(C)CC2CCCN2C(C2CCCS2)=O)cnn1C(C)(C)C 37544,C1(N(C(C2CC3(CSC3)C2)=O)Cc2ccc(C(F)(F)F)cc2)CCCCCC1O 37545,N1(C(C(C=C)O)=O)CC2CCC1CN2C(c1[nH]c(CC)cc1C)=O 37546,N(C1CCCc2cc(F)ccc21)C(c1cc2c(nc1)NC(=O)CO2)=O 37547,c1(-c2cn(CCCCCNC(c3c(C)cc(F)s3)=O)nn2)cccc(F)c1N 37548,C1(CNC(C(C)=C(C)C)=O)CCC(C)(C)CN1C(c1ccc(NC=O)cc1)=O 37549,C1(C(=O)NC2C(CNC(C(F)OC)=O)CCC2)CCC2CCCCC2C1 37550,c1(C(N2C(CNC(C(C)CSc3ccccc3)=O)CC2)=O)ccc(C2CC2)cn1 37551,C1(C(N2CCC(CC(C)NC(=O)CC3CCCCO3)CC2)=O)OCC2CCCC12 37552,CCC(CCOC)C(=O)N(CCNC(=O)C(C)(C)n1cccn1)CCOC 37553,CC1(C)CCCC(N2CCCC(Oc3ccc(C#N)cc3)C2)C1 37554,CCC(CC1CCCCC1)C(=O)NCC1CCN(C(c2ccnnc2)=O)C1 37555,C1(NC(=O)C(C2CC2)C2CC2)CCC2CCN(C(=O)C(O)c3ccsc3)C1C2 37556,n1(CC(N2C(CN(C(=O)C#CC3CCC3)C)COCC2)=O)ncc(C#N)c1N 37557,N1(C(Cc2c(C)nc[nH]2)=O)CC(NC(=O)Cc2cc[nH]c2)CC12CCCCCC2 37558,CCC(C)(CN)C(=O)NCC1(Cc2cc(F)ccc2F)CC(O)C1 37559,C(=O)(C(CNC(c1cc(C#N)n(C)n1)=O)C(C)C)N1CCC(CSC)C1 37560,C12(C(N3CC(C(C)NC(C(CC)(C)OC)=O)C3)=O)CCCC1C2(F)F 37561,CC1(C)CCCC(C(=O)NCCC2=CCN(C(c3ccc(C#N)[nH]3)=O)CC2)CC1 37562,c1(C(=O)NCC2(CCNC(C3CCCCO3)=O)CC2)cnc(O)c2ncccc12 37563,c1(C(N(CCCN(C(CC2CCC(C)O2)=O)C)C)=O)ncccc1Cl 37564,CCCC(CNC(c1scnc1C)=O)NC(=O)CSS(C)(=O)=O 37565,C(CS(=O)(=O)c1cccs1)NC(=NCC=C)NC(C)CNC(=O)OC(C)(C)C 37566,c1(C(N2C3CC(NC(C(CCC)OC)=O)C3CC2)=O)cccc2c1nnn2C 37567,N1(CCC)CCC(N(C)CC2(COC)CCC2)C1 37568,C(C(C(F)(F)F)N1CCN(C(c2cn(CC)nn2)=O)CC1)NC(CC=CC=C)=O 37569,C=CCC(F)(F)C(=O)NC1CCCC(NC(=O)Cc2ccc(Cl)c(F)c2)CC1 37570,C(CCCCC(=O)N1CCN(C(C2CC(C)C2)=O)C(n2ccnn2)C1)NC(C)=O 37571,C1(OCC)C(OCC)C2(C)CCC(C2)C(S(=O)(=O)C2OCCO2)C1(C)C 37572,c1(C(N(C(C)C(=O)NCc2ccoc2)CCC)=O)cc(CCOCC)on1 37573,c1(-c2cn(C3C(C(C)NC(=O)C4=CCCCO4)COC3)nn2)nccn2ccnc12 37574,CC1(c2cn(C3CCC4CC34)nn2)CCCO1 37575,c1(C(=O)NC(CNC(C2CC(OC)C2)=O)C)ccccc1C1(C#N)CC1 37576,C=CC1CCN(C(C2(CNC(=O)C(F)F)CC(=C)C2)=O)C1 37577,N1(CC(=O)N(Cc2scc(CNC(CCC(=C)Cl)=O)n2)CC)Cc2ccccc2C1 37578,C1(NC(c2cc(C)n(C(C)C)c2)=O)CN(C(C2CC2C2CCC2)=O)CC12CCC2 37579,C1(OC)CC(CNC(c2cc(C)nn2C2CC2)=O)N(C(c2cc(C)ccn2)=O)C1 37580,c1(OC)ccc(C(=O)NC2CC23CN(C(=O)OC(C)(C)C)C3)c(Cl)n1 37581,c1(C(=O)Nc2cccc(CNC(C(C)N(C)C)=O)c2)cc2c(cc1N)CCCC2 37582,c1(CC(=O)NC2(CC=C)CCN(C(=O)C(O)CF)C2)cn2cc(F)ccc2n1 37583,c1(C(N(CCOC)CCNC(c2cn(C)nc2C)=O)=O)ccc(OC)cc1C 37584,C1(C(=O)NCC2OCCCN(C(C3CC(=O)OC3)=O)C2)Cc2cncn2C(=O)N1 37585,C#Cc1ccc(CC(N2CCC(C(N3CC4CCCC3C4)=O)C2CC)=O)cc1 37586,C(=O)(C(C)(CC)CC)N(CC(CNC(C(CCC)=CCC)=O)O)C 37587,C(=O)(C(F)C(F)(F)F)N(C(C)C)CCOc1ccccc1F 37588,Fc1cc(Br)cc(NC2CCc3ccsc32)c1Cl 37589,CC1CN(C(c2cc(Br)ccn2)=O)CCN1C(=O)Cc1cnnn1C 37590,C12(F)CCC(C1)N2.c1(C(N(C)NC(C(C)OCC)=O)=O)ccc(C2(C)CC2)cc1 37591,c1(C(C(=O)NCC(C)N(C)C(C2(F)CCCCC2)=O)C)cncc(F)c1 37592,CC1OC2(CNC(=O)CC3CCCC(C)C3)CC1(NC(c1ccc[nH]1)=O)C2 37593,N1(C(C(C)SCC)=O)CCCC(CNC(C2CCCN2S(C)(=O)=O)=O)C1 37594,c1(OC)ccc(CC(C)(C)C(=O)NCc2ccc(Cl)cc2Cl)cc1OC 37595,CC(C)CC(CNC(c1csc(F)c1)=O)C(=O)NCCN1CCOCC1 37596,N1(C(C(C)NC(=O)OC)=O)CC2(CCCN(C(=O)CC3COCCN3C)C2)C1 37597,C(=O)(CS(=O)(=O)C1CCCC1)N(CCN(C(C(C)C1=CCCC1)=O)C)C 37598,Cc1cc(S(N)(=O)=O)oc1C(=O)NCCN(C(c1c(C)n[nH]c1C)=O)C1CC1 37599,N1(C(c2n(C)ncc2C#N)=O)CCC2(CC1)CCN(C(C1CC1CF)=O)C2 37600,c1(C(=O)NC2CN(C(C(C(=O)OCC)CC)=O)C2)cc(=O)n(C)c2ccccc12 37601,c1(CCC(N2CC(O)(CNC(c3ccc(F)nc3F)=O)C2)=O)c(Cl)cncc1Cl 37602,C1(C(=O)NCCC(C)NC(c2cnoc2C2CCOCC2)=O)CC(Cl)(Cl)C1 37603,Cc1cc(C(=O)N(CC(=O)NC(c2cnsc2)C)C)nc(C)c1 37604,C1(CNC(C2CN(C(=O)NC)C2)=O)CN(C(c2cc(O)ncc2F)=O)CC1(F)F 37605,C(=O)(C1=CC2C=CC1C2)NC(C(=O)NCCN(C(CC)C)C)(C)CSC 37606,Cc1nccc(C(N2CCCCC2CNC(C2(F)C(C)(C)C2(C)C)=O)=O)c1Cl 37607,c1(OC)nccc(CNC=O)n1.C1(NC(=O)CC2CCN(C)CC2)CCCCC1 37608,C1(C(N(C2CCN(C(c3nc(Cl)cs3)=O)C2)CCC)=O)CCC(C)(C)O1 37609,CCC(C(=O)N1CC(C(N)=O)(CNC(=O)CC2(O)CCOC2)C1)C(C)O 37610,C1(C(N2CC(OC)(CO)C2)=O)CN(C(=O)CC2CC=CCC2)CC1(F)F 37611,c1(CC(=O)NCC(C2CCC2)NC(C(C)OCC=C)=O)ccc(Br)s1 37612,C1(CNC(C2N(CC#C)CCC2)=O)CN(C(C2CSC(C)=N2)=O)CCC12CCC2 37613,c1(CC(=O)N(C(CNC(C(CC=C)C)=O)C2CC2)C)cnc2ccccc2c1 37614,c1(N2CCC(O)(C(C(=O)NC)(F)F)C2)cc(C)c(F)cc1[N+](=O)[O-] 37615,c1(C(NC(NCC(=C)C)=NCCC2CC2(Cl)Cl)C)ccc(C#N)cc1F 37616,Cc1nc(=N)[nH]c(C)c1C(=O)NCCC(C)NC(C1OC(C)CC1C)=O 37617,C1(C)(C(=O)NCC2(CC(=O)NC3(C(=O)OCC)CC3)CC2)C(C)(C)C1(C)C 37618,CC1=C(C(=O)NC2CC3CCC2N3C(=O)CC2(O)CCCCC2)CCO1 37619,C(CN=c1[nH]c(=NC2CC3CCCC3C2)c2ncccc2[nH]1)c1cccc(Br)c1 37620,N1(C(CCCCNC(=O)CC(=O)NC2CC2)=O)CC2CCCC(O)C2C1 37621,c1(CC)cc(C)c(C(=O)NNC(=O)C2CCCN(c3cc(O)ncn3)C2)o1 37622,C=CC1(CO)CCN(c2ncnc(NCCc3cc(C)ccc3Cl)c2C)CC1 37623,c1(OCC)nccc(C(=O)NC2CCCCN(C(C3CC=C(C)CC3)=O)C2)c1F 37624,c1(CC)cc(OC)ccc1C(N1CCC(CNC(c2c[nH]c(=N)o2)=O)C(C)C1)=O 37625,C(=O)(CCCCCNC(N)=O)N1CC(NC(C2(CC#C)CCOC2)=O)(CO)C1 37626,c1(N(CC(C2CCC2)NC(=O)OC(C)(C)C)C(C2CC(F)C2)=O)ccc(Cl)cc1 37627,c1(C(=O)NCC2OCC(CNC(c3ccc(O)nc3)=O)C2)ccc2nn[nH]c2n1 37628,c1(CN(C2CCN(Cc3cccc(C#C)c3)N(CC)C2)CCC)ccc2ccoc2c1 37629,c1(OC)ccc(CN2CC(N3CC(NC(=O)C(C)C4CC4)CC3=O)C2)c(C)c1 37630,c1(CS(N2CCC(CC(CC)OCC)CC2)(=O)=O)ccc(Br)c(OC)c1 37631,N1(C(C=CCC)=O)CC2CS(=O)(=O)CC2(NC(c2cc3c(cn2)OCCO3)=O)C1 37632,O=C(CCN=c1[nH]c(=NCCF)[nH]c2c1COC2)N1CCOCC1 37633,C(=O)(C1CCC(N)c2ccccc21)N1C(COC(C)(C)C)CCCC1 37634,C1(C(=O)NC2CC(C(=O)NCc3c(C)occ3)C2)CCC2(CCC2)C1 37635,N1(C(C=CCC)=O)CCN(C(=O)CC2C=NN(C)C2=O)CC1COC 37636,N12CCC13CCN(CC3)Cc1ccc(s1)NC(=O)C2=O.c1(C)cncc(Br)c1 37637,N1(C(CC=CC=C)=O)CCC2CC2(C(N2CC(OC(C)C)C2)=O)CC1 37638,C1(NC(c2c(-c3onc(C)n3)cccc2)=O)CN(C(C2(C)CCC2)=O)CC12CC2 37639,CC1(C)CCC(C(=O)NCC2=CCCOC2)(NC(=O)C=CCN2CCC2)C1 37640,c1(-c2cc(C(N(CCCNC(c3ccon3)=O)C)=O)no2)cccc(F)c1 37641,N1(C(CNC(=O)NC)=O)CC2(CC(NC(=O)C(C)CCCOC)C2)C1 37642,c1(C(N2CCC(CNC(c3ccn(C(C)C)n3)=O)CC2)=O)nccc(C#N)c1F 37643,C(=O)(CS(=O)(=O)C(C)C)N1CCN(C2CCCN(C(C(CCCC)C)=O)C2)CC1 37644,CCCCC(O)C(=O)N1CCC(CC(=O)Nc2nc(F)ccc2Br)C1 37645,N1(C(Cc2ccc(C)nc2)=O)CC2CC(NC(C3CCCC3N(C)C)=O)CC2C1 37646,c1(N(C)Cc2nncs2)[nH]c(=NCC2CC2C2CCC2)nc2scnc12 37647,N1(C(c2ccc(C(C)(C)O)nc2)C(=O)NC2CC2)CCC2(COC(=O)N2)C1 37648,C1(C)(C(c2nnnn2CSc2ccccc2)NC2C(C(C)C)C2)CCCC1 37649,N1(C(c2n(C=C)ncc2)=O)CCCC(NC(C2(c3ccccc3)CC2(F)F)=O)CC1 37650,C#CCCCCCCC(=O)N(CCCCCC(=O)NCc1cn(C)cn1)C 37651,c1(C(C)S(=O)Cc2coc(-c3ccc(Cl)cc3Cl)n2)ccc(F)cc1F 37652,c1(CC)cccc(F)c1C(=O)NCCC1CC(NC(=O)CC2(C)CCCC2)C1 37653,Cn1c(C(N2CCC(Cn3cc(C4(C(N)=O)CC4)nn3)C2)=O)cc2occc12 37654,c1(NC(C(=O)NCC(CC(C)C)C)=O)ccccc1S(C)(=O)=O 37655,N1(C(c2ccc(SC)o2)=O)CCCC(C2CN(C(c3cc(O)cc(O)n3)=O)C2)C1 37656,c1(C(=O)Nc2c(C(=O)NCc3n(C)ccn3)n[nH]c2)ccc(I)c(O)c1 37657,C1(CNC(c2c(C)nccc2)=O)C2CCC1CN(C(=O)C(C)C(C)(F)F)C2 37658,C(CC(F)F)(C(=O)NOCCC(C)O)N(C(=O)CC(C)(C)C(F)F)C 37659,c1(OC)cccc(C2CC2)c1.N12CCN(CC1)C(=O)Cn1cc(nn1)C2(C)C 37660,N1(C(CNC2C(C)(CO)CC2)=O)CC(O)C2CCCCC2C1 37661,c1(N(C(CNC(CN=[N+]=[N-])=O)=O)CC(F)F)cc(C(F)(F)F)ccc1C(F)(F)F 37662,c1(C(=O)NCC2CCCC2NC(C2CCOC2)=O)c[nH]c2ccccc12 37663,C1(C(=O)NCC2(NC(CNC(c3c(C)occ3)=O)=O)CCCC2)C2CC2C2CC12 37664,c1(OCC=C)ccc(C(N2CCOC(CCNC(=O)C=CC)C2)=O)cc1OCC 37665,c1(C(=O)NC(CC(C)NC(c2n(C=C)ncc2)=O)C)cc(Cl)c(N)c(Cl)c1 37666,C(=O)(CCCN=c1nccc[nH]1)NCCCN(C(=O)C1=CCCOCC1)C 37667,Cc1cc(F)c(C(=O)NC2(C3CCCN3C(=O)C(O)C(C)(C)C)CC2)cc1F 37668,n1(C(=O)NCC(COC)C(C)C)c(C2CC2)nc2ccccc12 37669,N1(C(CCc2ccc(C3C(C)C3)o2)=O)CCN(C(c2nc(C3CC3)cs2)=O)CC1 37670,O=C1OCc2cc(NC(C3CC34CCN(S(=O)(=O)C(F)(F)F)C4)=O)ccc21 37671,N1(C(c2c(OCC(=C)C)cccc2)=O)CCN(C(=O)CCCCC2CC2)C2CC12 37672,n1(NCc2cn(CC3C(OCC)CCC3)nc2)c(C(=O)O)nc2ccccc12 37673,c1(NC(C(C)C)=O)ccc(OCC(C)NC(=O)NCc2cnn(C)c2F)cc1 37674,N1(C(C(C(CC)C)O)=O)CCC2(CC1)CN(C(=O)COCCCOC)CC2CO 37675,c1(C(N2CCC(NC(c3c(N)cn(C)n3)=O)CC2)=O)cccc2ccccc12 37676,CS(=O)(=O)c1cc(C(=O)N=c2nc[nH]n2C2CCN(C(=O)OC(C)(C)C)C2)cs1 37677,C1(C(=O)OC)CCC(C(=O)NC(C)(C)C(C)NC(=O)CCCN(C)C(C)=O)CC1 37678,Cc1ccc(C=CC(N2CC(C(C)NC(c3cnn(CC(F)F)c3)=O)C2)=O)cc1 37679,c1(CC)c(C(N2CCC(C)C2C(=O)NCc2cnn(CC)c2C)=O)ccn1C 37680,c1(NC(=O)Nc2cc(OC)cc(Br)c2)ncc2ccccc2n1 37681,N(C1CCCn2ccnc21)C(C1(C)CCCN1C(=O)CC1(O)CCOCC1)=O 37682,c1(C(N2CCC(O)(CNC(C(CC)(C)CC)=O)C2)=O)noc(C)c1[N+](=O)[O-] 37683,C1(NC(c2ccco2)=O)CCC(n2cc(COCCNCCC#N)nn2)C1.C 37684,C(=O)(CCCC(=O)c1ccc(C)cc1)N(CC(CC)O)C1CC1 37685,CCC(O)CC(=O)N1CC(CCNC(=O)Cc2cccc(F)c2)C(C)C1 37686,O=C1NCCn2ncc(C(N3CC(CNC(C4CCC4(F)F)=O)C(O)C3)=O)c21 37687,C1(NC(C2N(C(c3c(OC)csc3)=O)CCC2C)=O)CC2(C1)CC(C)(C)C2 37688,S(=O)(=O)(c1ccc(N2CCC(CF)CC2)c(F)c1)N1CCSC(C)C1C 37689,C12(C(N(CCN(C(CC3C(C)=NNC3=O)=O)C)C)=O)CCCN(CCC1)C2 37690,C1(C(=O)NCCOC2CN(C(c3cc(CC)sn3)=O)C2)(OC)CCC(C)C1 37691,c1(C(N2CC(C)C(CNC(=O)CO)CC2)=O)c(Cl)ccc2ccoc12 37692,C(=O)(N=c1cc(Cl)cn[nH]1)c1ccc(CN(CCOC)Cc2ccc(F)cc2)o1 37693,Nc1cc(F)cnc1C(=O)NCC(O)CC(=O)NC(CC1CC1)C1CC1 37694,C(=O)(CC(CC#N)c1ccccc1)N1CCC(Cc2cn(C(C)CO)nn2)C1 37695,c1(OC)cc2c(cc1C(N1CCC(NC(=O)Cc3ccco3)C1)=O)OCO2 37696,C1(C2CC2)(CNC(c2cc(C)nc(O)n2)=O)CCN(C(=O)C(C)OC2COC2)C1 37697,CCC(C)(C)CCCC(=O)NC1CCC2CCN(C(=O)CCC(C)C)C12 37698,c1(C(N2CCC(C)C(N(C(=O)CC3CCCSC3)C)C2)=O)ccc(N=[N+]=[N-])cc1 37699,C1(CC(=O)N(C2CCN(C(C3C(C)C3)=O)CC2)CCO)COC2(CCC2)CO1 37700,c1(C(N2CC(O)(CCNC(c3cncc(CO)c3)=O)C2)=O)cnn2ccncc12 37701,c1(C(=O)NCC(F)CNC(C2(CC3CC3)CC2)=O)cnc(S)n1-c1ccccc1 37702,c1(C(=O)NC2C(C(=O)NC(C(=O)OC)CC(C)C)C2)cc(Cl)cc(Cl)c1[N+](=O)[O-] 37703,C(C(C(C)C)NC(C12CC(CO1)C2)=O)NC(C1C(C)C1C)=O 37704,c1(OC(c2c(Cl)cn(CC)n2)=O)cc(C)c(NC(C)=O)c(C)c1 37705,c1(CNC(C2CC(CC)C2)=O)nc(C(=O)N(CCCN=[N+]=[N-])C)c(C)o1 37706,c1(C(C)C)ccc2cc(C(N3CCC(O)(c4cnn[nH]4)C3)=O)ccc2c1 37707,CC(CN=C(NCc1cccs1)NCC1C(C)(C)C1(F)F)C(F)(F)F 37708,c1(C(c2ccc(-c3n(CCC)ncc3)s2)(C)C)ccc(O)cc1 37709,C(=O)(CCC(C)(C)N(C)C)NC1CC(N(C(c2c(C)nc(C(C)C)o2)=O)C)C1 37710,c1(C(N2CCN(C(C3C(OC)(OC)CC3)=O)C(CF)C2)=O)ccc2occc2c1 37711,N1(C(c2c(F)ncc(-c3cccc(C#N)c3)c2)=O)CCC2(CC1)CC(=O)NC2=O 37712,Cc1cscc1C(=O)NCC1(C(N2CCCC2C)=O)CC=CC1 37713,N1(C(c2c(C)onc2)=O)CCC2C(CCCN2C(=O)CN2CCC(C)(C)C2)C1 37714,c1(C(=O)NCCC(C)(C)NC(c2ccc(NC(C)=O)s2)=O)csc2nnsc12 37715,c1(OC)nc(N2CC3CN(C(=O)CCCCCCBr)C3C2)nc2[nH]cnc12 37716,C1(C(N2CC(OCCO)C2)=O)COCCN(C(c2cccc(O)n2)=O)C1 37717,C1(C(=O)NC2C3CN(C(c4nn(C)c(O)c4)=O)CC32)CC2(CCCC2)C1 37718,c1(C(N(C2CN(C(C3(C)CC=CCC3)=O)C2)C)=O)ccc(Br)cc1OC(F)F 37719,C1(NC(C=CCC)=O)CC12CCC(NC(c1ccc(C(F)F)o1)=O)CC2 37720,C1(NC(CN(CCC)C)=O)CCCC(NC(=O)C(C(C)CC)OCC)CC1 37721,C(C(C)(F)CNC(c1ccc(SC)o1)=O)NC(C(C1CC1)SC)=O 37722,C1(NC(c2nc(C(=O)OC)sc2)=O)CS(=O)(=O)CC1NC(c1cccc(Br)c1)=O 37723,c1(C(N2CC(CNC(c3ccnn3C3CC3)=O)C2)=O)conc1C1CC1 37724,c1(C(=O)NCC(C2CC2)NC(C2CC(C)(F)C2)=O)cc(F)cc2cc[nH]c12 37725,O=C(C#CC1CCCC1)NCCN(C1CCCC1)C(C12CCCC1CC(=O)C2)=O 37726,N1(C(C(C=C)(C)C)=O)CCC2(CC1)CC(CNC(c1cc(CO)[nH]n1)=O)C2 37727,C(C(O)C(C)(C)C)c1cn(C2(C(N(CC)CC3(O)CC(C(=O)O)C3)=O)CC2)nn1 37728,n1(CC(=O)NC2(CN(C(CSCC)=O)C)CC2)cc(C2CC2)nn1 37729,O=C(C1CSc2ccccc21)N1CC(Nc2nc(Cl)nc3sccc23)C1 37730,C(C#Cc1cn(CC2CCC2(F)F)nn1)NC(C1CCC(=O)N1)=O 37731,N1(C(C(CC)N2CCCC2)=O)CCN(C(=O)C(C)n2cccn2)CCC1C 37732,C(=O)(C(C)C(C)(C)C)NCCC1(OC)CN(C(c2n(CC)c(O)nc2)=O)C1 37733,N1(C(C(C)CF)=O)CC2CCC1C1CN(C(c3c(Br)nnn3C)=O)CC21 37734,C1(C)(NC(C(C(C)C)NC(c2sccc2C#N)=O)=O)CCC(=O)NC1=O 37735,C1(C(=O)NCC(C2CC2)SC)C2CC2CN1C(c1cnccn1)=O 37736,C1(NC(c2ccc(N)c(C)c2C)=O)CCN(C(=O)C2=CCCCC2)CC12CCC2 37737,c1(C(N(CCCNC(c2cccc(OCC)c2)=O)C(C)C)=O)cc2[nH]ccc2s1 37738,C(C(=O)NC1CCN(CCC(N)=O)CC1)(C(C(C)C)OC)OC 37739,C1(C(N(C)CC2N(C(Cn3c(C)ccn3)=O)CCCC2)=O)COC2COCC12 37740,C(=O)(CC(C)CC(C)(C)C)N1CC(c2cn(CC(=O)OC)nn2)CN(C)CC1 37741,c1(OC)cccc(C(=O)OC)c1-c1nc(CC(=O)OC)c(C)s1 37742,Cc1cccc2c1OC(C(=O)NCC(F)CNC(=O)CSCCC(F)(F)F)C2 37743,Cn1c(C(=O)NC(CNC(C2CCC(C(N)=O)O2)=O)C2CCC2)cccc1=O 37744,c1(C(=O)NC(C2(O)CN(C(CC(CC)C)=O)C2)C)cccc2nn(C)nc12 37745,C(=O)(CCCC(C)(C)C)NC(C)CC(C)NC(=O)C(C)(O)Cn1ccccc1=O 37746,C1(NC(=O)NC(c2cnn(C)c2)c2ccccc2)CCOC(C(F)(F)F)C1.CN1CC1 37747,N1(C(C(CCC)NC(C2CCOC2C(C)C)=O)=O)CCC(C)(CC)CC1 37748,C1(CC(=O)NC(C(=O)NCC(F)Cl)c2ccoc2)CCC(O)C1 37749,c1(C(=O)NCCCCCN(C(C(=Cc2ccco2)C)=O)C)nnc(S)n1C 37750,CC1(C)CC(C(=O)NC2CCC(CCNC(c3cc(C4CC4)no3)=O)C2)=NO1 37751,C1(C(=O)NCc2cnc(C)o2)CC(NC(=O)CCCn2cccn2)C12CCC2 37752,c1(NCC2CN(C(C3C(OCC)C3)=O)C2)cc(C(=O)OC)ncn1 37753,CS(=O)(=O)c1ccc(F)c(C(=O)NCC2(NC(=O)CC3CC=CC3)CCOC2)c1 37754,CCCCN=C(NCc1cc(OC)ccc1F)N1CCC(OC)C(C)(C)C1 37755,C1(S(N)(=O)=O)(C(N2CC(CC)C(NC(c3[nH]c(O)nc3C)=O)CC2)=O)CCCC1 37756,C=CCC(CC(C)C)C(=O)NC(Cc1cn(C2CCCC2)nn1)C(=O)OC 37757,c1(OC(C2C(C(=O)OCC)C2)=O)ccc(N2CCOCC2)cc1 37758,c1(C(N(CC(CNC(c2ccc(CC)cc2)=O)O)C)=O)c(Cl)cccc1[N+](=O)[O-] 37759,C(=O)(C1CSc2ccccc21)NC(CC)(C)CNC(=O)CC(C)(C)C(F)(F)F 37760,C(C)(N=c1[nH]c(=N)c2[nH]cc(Br)c2[nH]1)c1ccc(CC(=O)OC)cc1 37761,N1(C(C(=O)N(C)CC)C)CCOCC(C(=O)NCC(n2nc(C)cc2C)C)C1 37762,c1(CNc2nscc2C(=O)OCC2C(=C)C2)ccc2nc(O)n(C)c2c1 37763,CN1CC(C(=O)N2CCCC2CNC(=O)Cc2ccoc2)c2ccccc2C1=O 37764,C(=O)(C(O)CC[S+](C)C)N(CCCCCNC(c1cncc(OC(C)C)c1)=O)C 37765,CN=c1nc(C(N2CCCC(CNC(=O)CSc3ccccn3)C2)=O)cc(C)[nH]1 37766,C(=O)(C(C(=O)NCCCCC(=O)N(CC(O)CC)C)OC)OCC 37767,Cc1oc(C(N2CCOC(CCNC(C3CC3CF)=O)C2)=O)cc1Br 37768,C(C(CC(F)(F)F)NC(C1CCCN1N=O)=O)NC(Cc1n(C(C)C)cnn1)=O 37769,C1(OC(C(C)(CO)N(C)C)=O)C2CC3C1C3C2C(C1CCN(CC2CCC2)C1)=O 37770,CC1CC(NC(=O)C=Cc2ccc(C(F)F)o2)CN1C(c1ccc(C#N)o1)=O 37771,c1(CN(C(c2cscc2Br)C(=O)NCCC#N)C)ccc(S(C)=O)cc1 37772,C(=O)(CCC(CF)CF)N1CC(C)(C(=O)NC2(c3ccccc3)CC2)OCC1 37773,C(c1ccc(F)cc1)=CC(N1CCCN(C(=O)CC(O)c2ccccc2)CC1)=O 37774,c1(C(=O)NC(CNC(C(CCC)C)=O)CC)ccc2c(n1)NCCO2 37775,C1(CNC(C(C)NC(C)=O)=O)CCN(C(C2CC2C(C)O)=O)CC1C 37776,C1(C(=O)Nc2cccc(CO)n2)CCCC12CCN(Cc1cc(Cl)cnc1Br)C2 37777,Cc1nc(CCC(=O)NCC2CN(C(=O)C(C)OC3COC3)CC2C)[nH]c1C 37778,N1(C(CC=C)=O)CC(NC(c2ccc([N+](=O)[O-])cc2)=O)C(C2CC2)C1 37779,C1(COCC)CCN(C(C)C(=O)NCc2ncsc2C(F)(F)F)C1 37780,N1(C(CC2CC(C(C)C)OCC2)=O)CCC(CO)(NC(C2C3CCCC23)=O)CC1 37781,c1(C(C(=O)NCC(C2CC2)NC(Cc2cc(C(C)C)no2)=O)O)ccc(F)cc1 37782,C1(O)(c2cn(C(C)CNC(C3CCSC(C)(C)C3)=O)nn2)CCC(F)(F)CC1 37783,c1(CC(N2CC(NC(c3cccnn3)=O)C2)=O)c[nH]c2cc(Br)ccc12 37784,c1(OCC)nc(C(=O)NC2(C(=O)NC(CN(C)C)CCO)CC2(C)C)co1 37785,c1(C(N(CCCNC(C2CC2C)=O)CCC)=O)cc2n(n1)CCN(C)C2 37786,c1(N2CCC(C#N)C2)nc(N2CCC(C3CCCCO3)CC2)c2c(n1)CCS2 37787,c1(C(C(=O)Nc2ccccc2)N(CC(F)Br)C)cccc(Cl)c1Br 37788,N1(C(c2ccc(=N)[nH]c2)=O)C2CCC1(CNC(C1CCN(C3CC3)CC1)=O)CC2 37789,c1(CN2CC(NC(C3(F)CCCC=C3F)=O)C2)ccc2cc[nH]c2c1 37790,CCCC(C)CCCC(=O)NCCOCCNC(c1cn(CCO)nn1)=O 37791,Cc1ccc(C2CC2C(N2CC(CNC(=O)C(C)CF)C2)=O)cc1Br 37792,c1(C(N2C(C3CCN(C(C4CCN(C)C4)=O)C3)CCC2)=O)cc2c(F)cccc2[nH]1 37793,N1(C(C(C)=CC2CC2)=O)CCC(C(C)NC(=O)C(c2ncccc2F)(F)F)CC1 37794,c1(C(N(CC(CC)NC(=O)CCCNC(C)=O)C)=O)nccn2cnnc12 37795,N1(C(c2cc(C)on2)=O)CCCCC1CCCNC(c1cnc(O)o1)=O 37796,C1(NC(c2c(CNC(CCC(C)SC)=O)occ2)=O)CCC(C)(O)CC1 37797,C1(C(N(CCOCCN(C(C(C#C)(C)C)=O)C)C)=O)COC2(CCC2)CO1 37798,C1(C(N2CC(F)C(F)C2)=O)COC2(CCN(Cc3cncc(Cl)c3)CC2)C1 37799,Cn1nc(C2CC2)cc1C(F)(F)F.C12CCCC(C1)C(=O)NC(=O)C(=O)NC2 37800,c1(CCC(=O)NC23CC(NC(C4(COCC)CCCC4)=O)(C2)C3)cccc(C)c1 37801,c1(C(C(=O)NC(CC)C)N(C)C(C2(C)CC2)C)csnc1OC 37802,CC(C)CC(C(=O)N1CC2CC(NC(=O)CCC(C)(C)O)CC1C2)C(N)=O 37803,c1(SC)ncc(N)c(C(=O)NC(C)(CNC(=O)CN(C2CCSC2)C)C2CC2)n1 37804,C(=O)(C1=C2CCCN=CN2NN1)N1C2C(NC(C3CC3C(F)F)=O)CC(C2)C1 37805,C1(S(N)(=O)=O)(C=O)CCC1.c1(C(=O)NCC(C)(C)OCC)cn(CC(F)F)cn1 37806,C1(C(N2CCCC(CNC(C=C(COC)C)=O)C2)=O)C(O)C(=O)N(C)C1C 37807,N1(C(C2CC(F)(F)C2)=O)CCC(CCNC(C2COCCO2)=O)CC1 37808,CCCCCC(CC)C(=O)NCCCOCCC(N1CCN(C(C)C)C(=O)C1)=O 37809,Cc1ccccc1C(C)C(=O)NC1CCC(NC(=O)CCC2CCCCN2C)C1 37810,C1(CNC(CC2C(CNC(C3ON=C(C)C3)=O)C2)=O)CCC=CCC1 37811,N1(C(C(CCC)F)=O)CCCC(O)(CCNC(=O)CSc2nc(C)cc(C)n2)C1 37812,c1(C(C(=O)NC2CC(CNC(c3cn(C)nn3)=O)C2)O)ccc(Cl)cc1 37813,C1(CN(C)C(C2(F)CCOC2)=O)CCN(C(c2csc(-c3cn[nH]c3)n2)=O)CC1 37814,C(=O)(CC(C(C)CC)NC(=O)C(C)OC(C)(C)C)NC1(COC)CC1 37815,C=CCC(C)(CO)CN=c1[nH]c(N2CCC(C3CCC3)C2)nc2c1SCC2 37816,N1(C(C(C)OCCOC)=O)CCC2(CCC(CNC(C3CCCOC3)=O)CC2)CC1 37817,C1(O)(CNC(C(C)OCC2CC2)=O)CCN(C(c2nnn3c2CCC3)=O)CC1 37818,C1(CNC(C(c2ccc(F)cc2)C)=O)C(C)CCN1C(c1nnn(C)c1N)=O 37819,C(=O)(CCCC(=O)NCC(C)CNC(c1cc(C)nn1C)=O)NC 37820,Cc1cc(C(=O)NC2CN(C(=O)Cn3nc(Cl)ccc3=O)CC2O)ccc1Cl 37821,c1(C(N2C(CC(=O)Nc3cnn(C)c3C#N)CCC2)=O)cc2ccoc2cn1 37822,c1(C(=O)NCC(F)CNC(c2cc(Cl)c(Cl)[nH]2)=O)ccc(OCC(F)F)nc1 37823,c1(CC(=O)NCCN(C(C2CC2F)=O)C2CC2)c(F)cc(F)cc1F 37824,Cn1cncc(C(=O)NCCCN2CCN(C(=O)CCn3cccn3)CC2)c1=O 37825,CC1(OCCC(=O)NCCCOC2(CCCCO)CC2)CCC1 37826,c1(C(N2CCC(NC(c3cccn(C4CC4)c3=O)=O)C2)=O)ccn2ncccc12 37827,c1(C(CNC(=O)C(=O)N(CCC(C)N2CCCC2)C)OCC)cnc(Cl)s1 37828,C(C(=O)NCCC1CN(C(C2(C(F)F)CC(F)(F)C2)=O)CCO1)(C(C)C)OC 37829,C1(NC(=O)Cc2nccs2)CCC2CN(C(c3cccc(Cl)c3)=O)CC2C1 37830,C12(C(N3CC(NC(=O)NC)C3)=O)CCCC1C2 37831,C(CC(COC)(c1ccc(C)o1)NCc1nc(Br)ccn1)OC 37832,c1(-c2nc(-c3cc(Cl)ncc3)nn2CC2CCOC2)cc(F)cc(F)c1 37833,O=C1C(N2CCOCC2)CCCN1CCCc1ccc(O)cc1 37834,N1(CC2(C(C)C)CC2)CCN(CN(c2cccs2)C)CC1 37835,C1(NC(COCCC)=O)CC(F)(F)CC1NC(=O)C(C)Cc1ccc(OC)cc1 37836,c1(CC(=O)NC2CCCN(c3ccnc(Br)n3)C2)cnn2c1CCCC2 37837,C(=O)(CC(C)(C)c1ccc(F)cc1)NCC(N(C(C1(CC=C)CC1)=O)C)C1CC1 37838,c1(OC)ccc(C(=O)NCC2CCN(C(=O)C(O)C3CCCC3)CC2C)c(Cl)c1 37839,C12(C(N3CCN(C(c4cc(Br)c[nH]4)=O)CC3)=O)C3C4C1C1C2C3C41CO 37840,c1(C(=O)NC2(CNC(C(C)C3CC3)=O)CCC2)n[nH]c2c1COc1ccccc1-2 37841,C1(CC)(NC(=O)CC2CCCC2O)CN(C(C2CCC(C)O2)=O)C1 37842,CC(C)C(CCN(C(=O)C(C)C(F)F)C)NC(=O)Cc1ccc(Cl)cc1 37843,c1(C(C(=O)NCCOC)N(C2CCC(F)(F)C2)C)ccc(F)c(Br)n1 37844,Cc1ccc(C(=O)NCC2CCN2C(C2CCCC2C)=O)c(N)c1C 37845,c12ccnn1C(C)(C)NC2=O.C1(CC2C(C(=O)OC)C2)CCCC1 37846,N1(C(=O)CCC2CCCO2)CC2CCC(C1)N2C(=O)CC1CC2CC2C1 37847,N1(C(c2ccsc2C(F)(F)F)=O)CC2(C1)CN(C(c1ccnc(Cl)c1)=O)CCO2 37848,C1(C(N2C(CN(C(C(C=C)(C)O)=O)C)CC(F)C2)=O)C2CCC1(C)C2(C)C 37849,CC1C2C(CCN2C(C23CSCC2C3)=O)CN1C(=O)C=Cc1cc[nH]c1 37850,C1(CNC(c2c(OC)nn(C)c2)=O)CN(C)CCN1C(c1cc(N)cc(N)c1)=O 37851,c1(C(=O)NC2C(CNC(C(CCCC)O)=O)CC2)cc([N+](=O)[O-])ccc1O 37852,C1(NC(c2ncc(Cl)s2)=O)CCCC12CCN(C(c1ocnc1C1CC1)=O)CC2 37853,N1(C(=O)CN2CCOC2=O)CCN(C(=O)CC2CC23CC3)C(CCC(F)(F)F)C1 37854,c1(C(N2CC(NC(CCOCC(C)C)=O)C(C)CC2)=O)cc(Cl)cc2c1CCC2 37855,CS(=O)(=O)c1ccc(C(N2CCC(NC(=O)C(F)F)C2)=O)cc1Br 37856,c1(C(N2CC(CCn3cc(C4CCCO4)nn3)C2)=O)cnc(S)[nH]1 37857,C1(C(N2CC(CC(=O)NCc3nccc(OC)c3)OCC2)=O)CC(=O)OC1(C)C 37858,c1(CC(=O)NC2CC3(C(NC(C(CC#C)O)=O)C3)C2)ccc(Cl)cc1F 37859,C(=O)(C(CNC(=O)CN1CC(C)(C)C1)C(C)(C)C)NCCc1c(C)ncs1 37860,CCCCCCn1nnnc1C(C(C)C1CCC1)NCCc1cccnc1 37861,CC1CN(C(=O)CC2NC(=O)NC2=O)CC(C)CN1c1nnc(-c2ccon2)s1 37862,Cc1c(C(=O)NC(C)C(C)NC(c2c(Cl)ccc(Cl)c2O)=O)sc2ccccc12 37863,C(CC(=O)NCc1cccc(NC(=O)CC2CN(C(C)=O)C2)c1)(C(C)C)OC 37864,Cc1cc(C(=O)NC23CC(NC(=O)C(C)OCCC(C)C)(C2)C3)cc(C)c1N 37865,C1(CNC(CC(C)(C)SC)=O)CC12CCN(C(=O)Cc1cccnc1Cl)CC2 37866,c1(CC(=O)NCC2CN(C(C3CN(C4CCC4)C3)=O)CC2O)cccnc1Br 37867,C(=O)(C(F)(CC)C(=O)OC)N1CCC(NC(c2c(CCC)ccc(Cl)c2)=O)CC1 37868,c1(C(N2CCC(C)(NC(C3CCC(C)C3)=O)C2)=O)cc2c(s1)CN(C)CC2 37869,N1(C(CCCC(=C)C)=O)CCCC2(C1)CN(C(=O)CC1CCCCC1(F)F)C2 37870,c1(C(=O)NC(CC=C)CNC(=O)C(CC)N2CCCC2=O)ccc(Cl)cc1F 37871,N1(C(C2CC(C#C)(O)C2)=O)CCN(C(=O)CC2(CS(C)(=O)=O)CC2)CC1C 37872,Cc1nc2cc(C(=O)NC(C)CCNC(c3cccc4oncc34)=O)cnc2s1 37873,N1(C(CCC#C)=O)CCC(F)(F)C(C(=O)NC(C)(C)C#CCCC)C1 37874,c1(OC(C)C)ccc(Cl)cc1C(=O)N(CCC(C)NC(=O)CC1CC(CF)C1)C 37875,C1(C(=O)NCc2c(C)nc(CC)o2)CN(C(C2CC(C)(O)C2)=O)CCC1(C)C 37876,N1(C(C2CC(C)OCC2)=O)CCCCC2(CCOCC2)C1 37877,C1(C(N2C(CN(C(=O)CN3CCC3C)CC)CCC2)=O)CCC(C(N)=O)CC1 37878,c1(C2(CNC3CCC(C(=O)NCC4CCCCC4)OC3)CC2)cc(F)c(F)c(F)c1 37879,c1(C(N2CC(CNC(c3nc(C(C)=O)sc3)=O)C(C)C2)=O)c(C)nc(C)nc1C 37880,CC(CCC(=O)N1CC(n2cc(Sc3cccc(F)c3)nn2)C1)c1ccccc1 37881,C1(CNC(c2cc(C(N)=O)no2)=O)(CNC(=O)CC2CC23CC3)CC12CCC2 37882,c1(C(=O)NC2CC(NC(C(CC)n3ccnc3)=O)C2)n[nH]c(C)c1Cl 37883,Cc1cc(CC(=O)NC2CCCN(C(=O)C(=O)NCC(F)(F)F)C2C)ccc1F 37884,C1(C(N(CCC)CCO)=O)CN(C(=O)CC(C)C(C)C)CCC1(C)C 37885,C#CCC(C)C(=O)NCC1(O)CC(NC(C2CCCN(C(=O)C(F)(F)F)C2)=O)C1 37886,N1(c2cc(CC(C)C)ncn2)C2CCC1C(C)C(NC(C1CCC1)=O)C2 37887,c1(C(N2CCCN(C(C(=O)NCC)=O)CC2CO)=O)[nH]c2ccc(F)cc2c1C 37888,N1(C(c2nccc(OC)c2F)=O)Cc2cccc(Br)c2CC1C 37889,N1(C(=O)OCc2ccccc2)CCN(Cc2n[nH]cc2-c2ccc(Cl)cc2)CC1 37890,N1(CC(=O)NCCCC2(NC(C3CC3C(F)(F)F)=O)CC2)CCC(O)CC1 37891,N1(C(CCSCCCC)=O)CCC2(CCC2CNC(=O)CSC2CC2)CC1 37892,C1(NC(C(C)C(C)(F)F)=O)CN(C(=O)Cn2ccc(=N)[nH]2)CC2(CCC2)C1 37893,c1(C(N2CCC(CC(C)(C)C)C2(C)C)C(=O)NCC(=C)C)cc(Cl)c(Cl)c(Cl)c1 37894,C(=O)(C(C)(C)N1CCCC1)NCC(C)N(C(=O)CCNC(N)=O)C 37895,C1(C)(C(=O)NC2CCN(C(Cc3c(C(C)C)con3)=O)C2)CC(C(F)(F)F)=NO1 37896,C#CC1(NC(=O)C(CNC(c2ccnnc2)=O)C(C)(C)C)CCCCCC1 37897,C1(C)(C(=O)NCC2(OC)CN(C(=O)CC3CSCCO3)C2)CCN(C)C1=O 37898,c1(CC)ccc(C=CC(=O)NCCC(C)NC(=O)C=CCn2cncn2)o1 37899,N1(C(c2c(C)cc(Br)cc2)=O)CCC2CN(C3CCC3)CC2C1 37900,CCCS(=O)(=O)N=c1cc[nH]c(-c2ccc3nn(C)cc3c2)c1 37901,C1(NC(COCC(C)(C)C)=O)CN(C(C2CCOC(=O)CC2)=O)C(C)(C)C1 37902,c1(C(C)NC(C2N(C(c3c(C)nn(C)c3C)=O)CC2)=O)cccc2ccccc12 37903,c1(C(=O)NC2CN(C(CCCCC)=O)CC2C)ccc2c(c1)C(C)CO2 37904,C1(C(=O)NC(C)C(CO)NC(C2(N(C)C)CCCCC2)=O)CC(F)C(=O)N1 37905,C1(C(=O)NCCC(C(C)C)CO)CCCN1NC(=O)C1(C#N)CCOC1 37906,CCCC(C)(O)C(=O)NCC(CC1CC1)C(=O)NCC1CC(CC)C1 37907,C1(C(N(C2CCCOC2)CC)=O)C2CCC(C2)N1C(=O)CC1CC2C=CC1C2 37908,C(CS(=O)(=O)C1CCOCC1)NC(C(N)Cc1ccccc1F)=O 37909,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NCCCCN(C(C1CCC(C)CC1)=O)C 37910,N1(C(COCC#C)=O)CCN(C(=O)CC(C)COC)CC1Cc1ccccc1 37911,c1(C(=O)NC2C3CN(C(c4ccnc(O)c4Br)=O)CC23)ccn2ncnc2c1 37912,C1(C(=O)NCC2C(NC(c3ccc(CCC)[nH]3)=O)C2)CC(=O)N(CC(F)(F)F)C1 37913,N1(C(C(=O)N(C)C)=O)CC2(CCC2NC(=O)CC2CCCC23CC3)C1 37914,C(C)(c1cccs1)=CC(=O)NCC(c1ccc(F)cc1)NC(CCC)=O 37915,C(=O)(CC(F)(F)F)N(C1CCC(NC(=O)NCC2CN(C(C)=O)C2)C1)CC 37916,c1(CC(=O)NCCCN(C(=O)Cc2cnsc2)C)cccc2c1OC(F)(F)O2 37917,C1(NC(c2ccc3ccnn3c2)=O)CCN(C(c2cccc(F)n2)=O)C12CCC2 37918,C1(C2CCC2)(CNC(C2C3COCC23)=O)CCN(C(c2cccc[n+]2[O-])=O)CC1 37919,CC1CC(CCNC(C2(C)CC2)=O)CCN1C(=O)Cn1ncnn1 37920,CCC(CC(=O)N1CCCC(CCNC(C2(C3CC3)CCCO2)=O)C1)C(C)C 37921,N1(C(C(C(C)C)CNC(=O)CNC=O)=O)CCOCC(C)(F)C1 37922,N1(C(c2occ(C)c2C)=O)CCOC(C)(CNC(=O)CSCCC(C)C)C1 37923,C=CCCCCCCCCNC1(c2nnnn2CC(F)F)CCCC1CCCF 37924,c1(CC(=O)N(CC(C)CNC(=O)C=Cc2ncco2)C)cn2cc(F)ccc2n1 37925,C(=O)(C(O)C(F)F)NC1CC(NC(CN(CCOC)C)=O)C1 37926,c1(C(=O)NCC2CC(CNC(c3cc(Cl)no3)=O)C2)sc(F)cc1Cl 37927,C1(CNC(C(C(C)C)NC=O)=O)(NC(=O)CC2CC2(Cl)Cl)CCCCCC1 37928,c1(C(=O)NCC2CC(NC(C3CCCC3COCC)=O)C2)cccc(C#N)c1C 37929,C1(C(N)=O)(SC)CN(C(C2(CCNC(C3CC3(Cl)Cl)=O)CC2)=O)C1 37930,c1(SCC(N2CC(NC(c3cc(C)oc3C)=O)C(O)CC2)=O)ccc2c(c1)CCC2 37931,c1(NC)c(C(=O)NCC(CO)NC(=O)Cc2ccc(Cl)nc2)sc2nccnc12 37932,C1(CC)CN(C)CCCN1C(C1CN(C(C2CCC3(CC2)CC3)=O)CC12CC2)=O 37933,c1(C(N2CCC(C(C)NC(C3C(C(C)=O)C3(C)C)=O)CC2)=O)ncnc(C)c1C 37934,CC(C)(C)CC(O)C(=O)NCC1CC(CNC(=O)CNc2nccs2)C1 37935,C(=O)(C1COc2ccccc21)N(CC)CC1CCN(C(=O)CC(C)F)CC1 37936,c1(C(=O)NCCNC(CC2(CSC)CC2)=O)nnn(C)c1C.C1(SC)CCCCO1 37937,c1(C(N2CC(NC(C(CC)OC)=O)C2)=O)ccc(OC(C)(C)C)cn1 37938,Cc1ccc(C(N2CC=CC(NC(C3(C)CCCS3)=O)C2)=O)c(N)c1F 37939,CC1(CNC(=O)CCN2CCCCC2=O)CCCN(C(=O)Cn2cnnc2)C1 37940,C(C)(CN=c1[nH]nc(C(C)C)o1)NC(c1n(CC)nc(C(C)C)c1)=O 37941,n1(CC(=O)N(CC)CC)nc(C)c(-c2cscn2)c1C 37942,C(C)(CC(=O)NCCCC1(O)CC1)NC(C1(OC)CC1)=O 37943,c1(CC(=O)N(C2CCCCN(C(=O)C(O)C3CC3)C2)C)ccc2occc2c1 37944,c1(-c2c(C(=O)NCC3C(NC(CC(=O)OCC)=O)C3)c[nH]n2)ccccc1Cl 37945,Cc1nc2sccn2c1C(N1CCC(NC(=O)CC2CC2(Cl)Cl)C12CC2)=O 37946,C1(CCNC(C=CC(=O)OCC)=O)CSCCN1C(=O)CS(=O)(=O)NC 37947,c1(C(=O)NCC(C(C)C)NC(=O)C(C)Cc2cccc(F)c2)ncc[nH]c1=O 37948,c1(NCc2n(CC(=O)OC)ncc2)ccc2c(c1)CCC(C)C2 37949,Cc1cc(C(=O)NC2CC2NC(=O)Cn2cnc(=N)[nH]2)c2c(Br)cccc2n1 37950,C1(CNC(CN(C)CC)=O)CCC(CNC(C2CCCN(C(=O)NC)C2)=O)CC1 37951,C1(C(=O)NC(CCCC)CNC(=O)CNC(=O)CN(C)C)CC(=O)NC(=O)N1 37952,c1(C(=O)NCc2ccc(-c3cnc(O)nc3O)nc2)ccc(I)cc1[N+](=O)[O-] 37953,c1(OC(C)C)ccc(CN2CCC(O)C(C(=O)NCc3cnn(C)c3)C2)c(Cl)c1 37954,Cc1cc(CN(C)C(C2C=CCCN2C(C2CC2Cl)=O)=O)n(C)n1 37955,Cc1cc(C(N2CCOCC2C(N2CCOCC(O)C2)=O)=O)cnc1C 37956,c1(CC(C(=O)N(C)CC2(CNC(C3(OC)CC3)=O)CC2)C)c(C)nn(C)c1C 37957,c1(C(=O)NC(CNC(CCc2ccnc(C)n2)=O)C)cn(C2CC2)c(C)cc1=O 37958,CC(C)(C)C(C(=O)NC12CCN(C(=O)COC3CCCC3)CC1C2)NC=O 37959,CC#CCCCC(=O)N(CC(C)CNC(=O)C(C1CCOCC1)C)C 37960,C(C)(C(=O)N1CC(CN(C(=O)Cc2ccc(F)nc2)C)C2(CC2)C1)(C(C)C)OC 37961,C(=O)(CCC(=O)C(C)(C)C)OC.n12cc(nn1)CC1CN(C1)C(=O)C2 37962,N1(C(C(C)OC)=O)CCC(CCC(=O)NCC(C)CCO)C1 37963,N1(C(C(c2cnn(C)c2)OC)=O)CC(C)(CNC(=O)CCCCSC)CC1(C)C 37964,CC(C)CCC(O)C(=O)NC(CC1CCC1)C(=O)NCc1cccnc1Cl 37965,S(=O)(=O)(c1ccc(NCc2ccncn2)c(Cl)c1)NCC(C)(C)CCCO 37966,c1(NCC(=O)NCC2(O)C(C)OCC2)ccc(=O)n(-c2ccncc2)n1 37967,Cc1ccc(NC(C2(NC(=O)CN3CC4CCC3C4)CCOCC2)=O)cc1C 37968,c1(C(=O)NC2CCN(C(C(n3ccc(Br)n3)C)=O)C2)ccc2ccccc2n1 37969,CC(C)C(C)(C)C(=O)NC1CC(NC(c2c[nH]nc2[N+](=O)[O-])=O)CC1O 37970,c1(N(C)Cc2ccc(CC)s2)nnc(-c2oc(C)nc2C)n1CCCn1cnnn1 37971,C(=O)(C(CC(C)C)NC(=O)CCCC1(OC)CCC1)N1C(CC(=O)OCC)CC1 37972,c1(C(=O)NCC(CCCC)NC(C2(CC#C)CC=CCC2)=O)cc(F)ccc1N 37973,c1(C(=O)NC2C3(CC(NC(C(CCSC)O)=O)C3)C2)cc(Cl)ccc1O 37974,Cc1cnc(N2CCOCC(C(=O)NC(C)CCO)C2)nc1N1CC(C)OC(C)C1 37975,C(=O)(CC(CN(C)C)CC)NCC(CC)NC(c1ccc(CO)o1)=O 37976,c1(C(C)OC)nc(N2CCC(CNC(C3CCC(N=[N+]=[N-])C3)=O)C2)cc(Cl)n1 37977,C(=O)(CN=c1cc[nH]cc1)N1CC(CC(N2Cc3c[nH]nc3C2)=O)OCC1 37978,N1(c2ncc(C(=O)OC)nc2)CCC2(CCCN(C(=O)CC3(O)CCOC3)C2)C1 37979,CCCCC(CNC(=O)COCCCOC)NC(C1CCS(=O)(=O)C1)=O 37980,CCC(CN(C)C)CC(=O)N1CC2(C1)CN(C(=O)Cc1nc[nH]n1)C2 37981,c1(C(N2CCC(O)(CN(C)C(c3cc(F)n[nH]3)=O)C2)=O)[nH]c2ccccc2c1Cl 37982,C=CC1(C(=O)NC(C)(C=C)CC)CCN(C(=O)C(O)C=C)CC1 37983,C12(C(=O)NCC3CN(C(c4cccc(N)c4)=O)C3)CC1Cc1c[nH]nc12 37984,CC1(C)CCOC(C(=O)NCC2CCCCC2C(=O)NCc2ccc(O)cc2)C1 37985,C1(CCC)CN(C(c2cc(N)ccn2)=O)CC1NC(=O)C(CSC)OC 37986,N(C(=NCCC(=O)NC)NC1CCN(CC2CCCC2)C1)C(c1nnc(C)s1)C 37987,c1(C(N(C)CC)=O)cccc(C(=O)NCC2CN(C(=O)C(C)COC)CCO2)c1 37988,CCCCCC(C)NC(=O)CC1CCC(NC(=O)CCCC2CCCC2)CC1 37989,C(=O)(C1=CCCC1(C)C)NC(C(C)C)(C)CNC(=O)CCOCC1CCCO1 37990,c1(C(N2CC(NC(c3ccc(SC)cc3)=O)C(F)C2)=O)cccc2nccnc12 37991,C(=O)(C1CCc2c[nH]nc21)N(C1CCCN(C(=O)CCc2cccs2)C1)CCO 37992,c1(C(=O)NC(c2cn(CC3CC=CCC3)nn2)CCC)cc2nccn2c(O)n1 37993,N1(C(C2(C=C)CCCC2)=O)CCN(C(=O)C(O)C(F)(F)F)CC1C 37994,c1(CC2OCCN(Cc3c(C)n(C)nc3)C2)ccc(F)cc1F.C1(=O)CN1 37995,C1(C(=O)NCCCCNC(Cc2ccc(C)o2)=O)CCn2nncc2C1 37996,c1(C(N2CC3(OCC(NC(CCC=C=C)=O)C3)C2)=O)cc(C)c2c(c1)CCC2 37997,CN1CCc2c(C(N3CCCC3C(=O)NC3CC(F)(F)C3)=O)cccc21 37998,c1(C(=O)NC23COC(CNC(C4(CF)CC4(F)F)=O)(C2)C3)cn2c(n1)CCCC2 37999,N1(C(CSCCN(C)C)=O)CCC(N(C)C)(CNC(C2CCCSC2)=O)C1 38000,c1(CC)ccc(C(=O)NC(C)CNC(=O)CCC2CCOCC2)cc1S(C)(=O)=O 38001,c1(C(=O)NC(C2CCN(C(CSCC)=O)C2)C)cccc(Br)c1 38002,C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CCC(C(=O)Nc2ccc(C=C)cc2)CC1 38003,c1(CC)cc(=NC(=O)C(CNC(C2(CC)CCC2)=O)CC(C)C)[nH]n1C 38004,C(=O)(C(=NOC)c1ccco1)NC1CCCCN(C(C2C(C(=O)OC)C2)=O)C1 38005,N1(C(C(C)OCCC)=O)CCN(C(=O)C(c2ccccc2)O)CC12CC2 38006,N1(C(C(CC)CO)=O)CC2(CCC(NC(c3cc(OC)cs3)=O)CC2)C1 38007,c1(CCN(C)CC2CCCN2C(C2(O)CC3CCC2C3)=O)c(F)cccc1F 38008,c1(C(=O)NC2CCCC(C(=O)N(C3CCOCC3)CC)C2)ccc2c(c1)CCCS2 38009,c1(CC(N2CCCCC(NC(C3CCCS3)=O)C2)=O)cnc2cccnn12 38010,c1(C(C)(C)C)nc(C(=O)NCC2CCCC2)n[nH]1.C(=O)(C(F)=C1CCCC1)N 38011,C1(C(=O)NC2CON(CC)C2=O)(NC(C(C)OCC#C)=O)CCCCC1 38012,c1(C(=O)NCC2N(C(CC=CC=C)=O)CCC2)cc2c(OC(F)F)cccc2[nH]1 38013,N1(C(c2n(C)ncc2)=O)CCC2CCC12CNC(=O)CNc1cccc(Cl)c1 38014,N1(C(c2cccc(C)c2O)=O)CC(N=[N+]=[N-])CC1C(=O)NCC(O)C(N)=O 38015,c1(C(=O)NCC2CCC(OC)(OC)CC2)nccc2ccc(Br)cc12 38016,Cc1cc(Cl)c(C(=O)NNC(=O)C2CCN2S(C)(=O)=O)c(Cl)c1 38017,C(=O)(C(C)(C)CO)NC(c1n(C)ccn1)c1ccccc1 38018,CC(C(=O)NCCC1CCN(C(c2ccc(C(F)F)cc2)=O)C1)C(F)F 38019,C12(NC(C3(CC)CC3)=O)CC1CN(C(C1(CN(C)C)CCCC1)=O)C2 38020,N1(C(CC2CC(OC)C2)=O)CCCC(F)(CNC(=O)C(C)(C)c2ccccc2)C1 38021,c1(CCNC(CC2CCC(C(CC)(C)C)CC2)=O)cnc2c(Cl)cnn2c1 38022,N1(C(C2N(C)CCC2)=O)CCC(C)(C)C1CC(N1CCC1CN=[N+]=[N-])=O 38023,Cc1cc(C(F)F)n(CC(N2CCCCC2C(C)NC(=O)C(C)(C)CO)=O)n1 38024,N1(C(CC2CC(CC)C2)=O)CCC2CCCC12CNC(c1ccnc(Cl)c1N)=O 38025,c1(C(N2CCC(O)(CNC(c3cc(SC)c(C)o3)=O)C2)=O)ccc(N)c(Cl)c1O 38026,C1(NC(C2C(C)(C)C2)=O)CCC2CN(C(C34C5C6C3C3C4C5C63C(N)=O)=O)CC12 38027,c1(CNC(C(c2cn(C)nc2)=O)=O)ncccc1C(=O)NC1CCCOC1 38028,CCCCCCCC(=O)N1CC(CC(=O)NCCCCN(C)C)C2(CC2)C1 38029,C1(C(C)C)CCC(C(=O)NC(C2CN(C(c3ccc(C4CC4)o3)=O)C2)C)CC1 38030,c1(C(=O)NC2CCN(C(C3(N(C)C)CC3)=O)CC2O)c[nH]c2cc(C#N)ccc12 38031,C1(NC(c2ccc(O)cc2)=O)CN(C(C2CC2CF)=O)C2(CCCC2)C1 38032,C1(C)(CC)CC(C(=O)NC(Cc2ccoc2)CO)CCO1 38033,C1(OC)CN(C(=O)Cn2nccn2)C(C)(CNC(c2ncc[nH]c2=O)=O)C1 38034,CC(C)(C)C(C(=O)NCCC1CC(NC(=O)CCn2cncn2)C1)n1ccnn1 38035,C12(CCNC(C(C)N(C)C(C3CCCC3C(=O)OC)=O)=O)CC(CO1)C2 38036,c1(C(=O)NCCC2N(C(c3ncn(C)c3)=O)CCC2)cnn(C)c1S(C)(=O)=O 38037,N1(C(CC(C)O)=O)CC2CCC(C1)C(NC(C1(c3ccnn3C)CC1)=O)C2 38038,c1(C(N2CCC(CCCNC(C3SC4C=CC3C4)=O)CC2)=O)cccnc1CO 38039,c1(C(N2C(C(=O)OC)CC2C)C(=O)NC2CCCC2)nc2cc(Br)ccc2s1 38040,C(C1CC1)(C1CC1)=CC(=O)NCCCN(C(c1cc(SC)oc1C)=O)CC 38041,C1(CC)CCCCC1C(N1CC(C(C(=O)NC(c2ccn(C)n2)(C)C)OC)C1)=O 38042,c1(C(N2CCC(COC)(NC(c3cnc(O)n3C)=O)C2)=O)c(C)nn(C)c1OC 38043,C=CC1CN(C(C2(N(C)C)CC2)=O)CC1NC(=O)CNC(=O)CCC 38044,N1(C(C2(C#N)CC=CC2)=O)CCC(NC(c2ccc(Cl)nn2)=O)C(CO)CC1 38045,C(=O)(CCCCC(F)(F)F)NC1CC(NC(C=C2CCC(C)C2)=O)C1 38046,c1(C(=O)NCC(C)NC(C(CCCC=C)(C)C)=O)ccc2c(c1)NC(=O)CCC2 38047,N1(C(=O)CSc2cn[nH]c2)CCC2CN(C(C3Cc4nccn4C3)=O)C2C1 38048,N1(C(C#CCNC(C(CC2CCC2)OC)=O)=O)CC(F)(F)CC1C 38049,N1(C(c2c(C(C)C)scn2)=O)CCC(CNC(c2cc(N)c(F)cn2)=O)C(C)C1 38050,c1(C(=O)NC2(C)CC(NC(c3cccnc3O)=O)C2)cc2c(s1)CCOC2 38051,N#CC1(CC(=O)NC2CCCCN(C(=O)CN3CCNC(=O)C3)C2)CCOCC1 38052,C12(C(=O)NCCC(C)NC(=O)CC3CC4(COC4)C3)CCC(CC1=O)C2 38053,N1(C(CCCC2C(C)C2)=O)CCCN(C(c2cc(O)nn2C)=O)CC1C 38054,c1(C(=O)NC2CN(C(C)C)C(=O)C2)ccc2c(c1)CCN(C(=O)Cn1ccnc1)C2 38055,C12(NC(=O)CCSC(F)(F)F)CCCN(C(c3ccc(F)o3)=O)CC1C2 38056,CC1CN(C(=O)Cc2cnoc2)CC(CCNC(=O)Cc2cnn(C(F)F)c2)O1 38057,c1(CNC2CCC(C(N3CCC(C#N)C3)=O)CC2)c(F)cc(Cl)cc1Cl 38058,c1(N2CCOCC(NC(c3cnn(CC)n3)=O)C2)ncc(Br)cc1C#N 38059,C(=O)(C(CC)C(C)C)NCC1(O)CC(NC(C=CC=CC)=O)C1 38060,Cc1cc(Cl)cc(C(N2CCCCC2CNC(=O)CC2CCCOCC2)=O)c1N 38061,c1(C(=O)NCC(CNC(c2cn(-c3cccnc3)nn2)=O)OC)ncccc1Cl 38062,C1(COC(C2CCC(c3ccccc3)O2)=O)CCCCC1N1CCCC1=O 38063,CCC(C)C(C)CN=c1[nH]c(=NCCCc2nc(C)cs2)c2cc(Cl)ccc2[nH]1 38064,c1(C(=O)NC(C2(O)CCCCC2)C(=O)NCCCCN(C)C)cc([N+](=O)[O-])n[nH]1 38065,C1(C(N(CCCN(CC(=O)NCCOC(N)=O)CC)C)=O)CC1(C)CC 38066,C1(C)(CNCc2nc(C)n(C)c2C)CCCC(C)(C)C1 38067,N1(C(=O)CC2CC3CC3C2)CCN(C(c2cnc(C3CCC3)o2)=O)C(CCO)C1 38068,c1(C(=O)NC2CC(NC(C3(C)CCC(C)CC3)=O)C(O)C2)cc(C#N)ccc1O 38069,CCCCCC(O)CC(=O)NC1CCC(CNC(=O)CCCN(C)C(=O)OC)C1 38070,CC(C)(C)C(C(=O)NNC(=O)C1CN(S(=O)(=O)c2ccccc2)C1)c1ccccc1 38071,C1(NC(C(CC=CC)C)=O)Cc2ccccc2C1NC(=O)CCc1cnoc1 38072,CCCN=C(NCCN1CCN(C)CC1c1ccccc1)NC1CC(CC)C1 38073,n1(CCC(=O)NCC2C=CC(NC(C3C(C=C)C3)=O)C2)ccccc1=O 38074,C(=O)(C1=CCCC1(C)C)NC(C(C)(C)NC(CC1(C=C)CCC1)=O)C 38075,N1(C(CC2CCN(C)C2)=O)CCC2(CCCC2CNC(=O)CC2CCC2)CC1 38076,N1(C(C2(C)CC2(F)Cl)=O)CC2CCC(C1)N2C(c1cnns1)=O 38077,N1(C(COC(C)(C)C)=O)CCC2(C1)CN(C(=O)CC(F)(F)Br)CCO2 38078,Cc1nc(-c2ccccc2Oc2ccc(-c3nn[nH]n3)cc2)n(C2CCOC2)n1 38079,CC1COC(C)(C)CN1C(=O)NC(c1cccnc1Br)C 38080,C1(CC)CN(C(=O)CO)CCC1NC(=O)C(N1CCCCCC1)c1ccc(F)cc1 38081,c1(N(CCC#N)C)cccc(C)c1.c1(CCC)cnc(CN)s1 38082,c1(N2CC(C)(NC(c3ccc(C#C)cc3)=O)C2)nc(CC)nc2sccc12 38083,C(=O)(C(O)C(C)(C)C)NC1CC(C)(NC(c2nc(CN3CCOCC3)cs2)=O)C1 38084,C#CCCCCCCCNC(=O)CC(CC)NC(c1cc(C)cc(C)c1)=O 38085,Cc1ccnc(F)c1NC(=O)NCCc1ccc(Br)cc1C(C)C 38086,C12(C(CNC(c3cn(C(F)F)cn3)=O)NC(c3ccoc3Cl)=O)CCC(CC1)C2 38087,O=C(C(CO)c1nn[nH]n1)NCC1CC(Cl)(Cl)C1 38088,N1(C(c2cccc(Br)c2)C)C2CCCC1CN(C(C1(C)CC1)=O)C2 38089,N#Cc1c(N2CC(C3(NC(=O)CCC4CCC(C(N)=O)O4)CC3)C2)cccc1F 38090,N1(C(c2cncc(OC(C)C)c2)=O)CCC(C2(O)CN(S(=O)(=O)C3CC3)C2)CC1 38091,CCCCC(C)CCC(=O)N(CC(C)O)CCNC(c1cccc(C)c1N)=O 38092,c1(C(N2CCC(NC(C3(CC#C)CC3)=O)C(O)C2)=O)ccc2nc(C)[nH]c2c1 38093,Cc1c(C(=O)NC2(C)CCN(C(=O)C(C)O)CC2)sc2[nH]cnc(=O)c12 38094,C1(NC(C2C(OCC)C2C)=O)CCS(=O)(=O)C12CN(C(=O)Cn1cc(CO)nn1)C2 38095,C(C)(C(C(=O)NC1CC(O)C1O)NC(C1OCCC1(C)C)=O)OC 38096,C1(NC(C2C(C)N(C(=O)CCc3csnn3)CC2)=O)CCn2nnnc2C1 38097,N1(C(C2=CC(C)(CC)C2)=O)CCCC2(NC(=O)C(F)=C(C)C3CC3)CCCC12 38098,Cc1nn(C)nc1C(=O)NCC1(CNC(c2cc(Cl)cs2)=O)CCCC1 38099,O=S(=O)(c1cnc(Cl)c(NCCC2CC2(Cl)Cl)c1)N1CCN(CC(F)(F)F)CC1 38100,c1(OC(C)=O)cccc(-c2cc(NC(=O)Cn3cc(Cl)cn3)ccn2)c1 38101,Cc1[nH]c(CN2CC3CC2C3C(=O)Nc2ccc(Br)c(Cl)c2C)c(C)c1[N+](=O)[O-] 38102,CCC(C)CC(C)C(=O)NCC1CC2CCC1N(C(c1cnnc(Cl)c1)=O)C2 38103,C1(C)(C(=O)NC(CCOC)C(N)=O)CCCN(C(c2ccco2)=O)C1 38104,N1(C(CC=CC=C)=O)CCC(NC(=O)CC(C)COC)C1C 38105,N1(C(c2cc(OC(C)C)ncc2)=O)CCC(C)N(C(=O)C(O)C(C)C)CC1 38106,C1(C(=O)NCCCC(C)NC(c2ccnn2CC2CCC2)=O)CC2CCC1CC2 38107,C(C)(C(=O)NC1CCCC1NC(=O)Cc1ccoc1)(C1CCOCC1)NC(C)=O 38108,C1(CC)(NC(=O)C(C2CCCCC2)F)CN(C(=O)C(C)COC)C1 38109,c1(CC)c(C(=O)NCC(C)(C#N)CO)cnn1C(C)(C)C 38110,c1(OC)cnc(C(=O)NC2(C)CC(NC(c3n[nH]c(C4CC4)n3)=O)C2)c(F)c1 38111,C1(Nc2ccc(C(C)=O)cn2)CCN(C(c2cnn(C(C)(C)C)c2)=O)C(C)C1 38112,C#Cc1ccc(C(=O)NC2C3CC2N(C(=O)CC2CCC(C)C(C)C2)C3)nc1 38113,C(=O)(CCCCc1cn(C2CCC(C(=O)N(C3CCNC3=O)C)C2)nn1)OCC 38114,C1(C(=O)NC2CN(C(C34CC(C3)C4)=O)CCC2C(F)(F)F)CCc2nc[nH]c2C1 38115,c1(OC(C)C)ncc(C(=O)NCCCNC(c2ccc(CO)cc2)=O)cc1Cl 38116,c1(CC(N2C(C)(C(=O)NCC(C)OCC=C)CC2)=O)ccc(C)c(C)c1 38117,C(=O)(CCN(OC)C(=O)CCCCCNC(=O)CC1CCCC2CC12)OC 38118,c1(C(=O)NC2(C)CC(C(N(CC(C)SC)C)=O)C2)cccc(F)c1F 38119,c1(C(=O)NCCN(C(C(C)C2CCCO2)=O)C2CC2)cnc2sccc2c1 38120,C1(CNC(C2(CC#C)CCCO2)=O)CC(C)CN(C(=O)C(OC)OC)C1 38121,c1(CCNC(C)(C)C)cc(C(=O)CCN(C(=O)OC2CCCCC2)CCO)no1 38122,C(CCC(CO)NC(=O)CCNC(C)=O)NC(c1c(CC)nc[nH]1)=O 38123,c1(C(N(C(CNC(c2ccc(C)nc2O)=O)C2CC2)C)=O)c(Cl)ccc(F)c1C 38124,C1(NC(c2cc(C)nc(O)c2)=O)CC2CC1CN(C(C1CCC(F)C1)=O)C2 38125,C(=O)(C(O)CC(C)(C)C)NCCCC(CCC)NC(C1CS(=O)(=O)C1)=O 38126,C(N=c1cc2c(c[nH]1)CCCC2)c1cc(C(=O)OCC)c(OC2CC2)cc1 38127,c1(C(=O)NC(C(C)(C)NC(C(CCSC)O)=O)C)ccc(C2=NOC(=O)C2)cc1 38128,CCCCC1N=C2C=CN(N2)C2NCCN(C1=O)CC2 38129,c1(C(N2CC3CN(Cc4c(OC)nccc4)C3C2)=O)cc(C)c(Cl)cc1Cl 38130,C(=O)(C1CCCc2n[nH]cc21)NCC1(NC(=O)Cn2cccc2)CC(OC)C1 38131,c1(C(N(C2CCN(C(c3cncs3)=O)C2)CC)=O)cc2cccc(F)c2s1 38132,c1(OCC=CC)cccc(CC(=O)NC2CCCN(C(=O)CC34CC(C3)C4)C2)c1 38133,C1(NC(c2cc(-c3cccnc3)no2)=O)CC(F)CN(C(C2CCCSC2)=O)C1 38134,C=CCCCC(C)(C)C(=O)N1CC(CC(C)(C)CNC(=O)COC2CCCOC2)C1 38135,CS(=O)(=O)c1cccnc1C(=O)NCC1CCC2C(C1)C2(F)F 38136,N1(C(C)=O)CCC2CN(C(=O)C(C)(C)c3cscc3Cl)CCC2C1 38137,c1(N2CCC3(C(C(=O)NC(c4nc(=O)o[nH]4)C)C3)CC2)nc2ccc(Cl)cc2s1 38138,N1(C(C2N(C(C(C)C)=O)CCC2)=O)CCN(C(C2CCCS2)=O)C2(CC2)C1 38139,c1(CC(=O)NC(C)CNC(=O)CCc2ccccc2O)ccc(Cl)nc1F 38140,Cc1cnnc(C(=O)NC(C2(O)CN(C(c3ccc(C(C)C)cn3)=O)C2)C)c1 38141,Cn1nc2c(c1-c1cncnc1C(=O)Nc1cc(O)ccc1Cl)CCC2 38142,C1(NC(NC2C(CC=C)CCCC2)=NCCC)(C(=O)OC)CC2(CC(F)C2)C1 38143,CCCCC(F)C(=O)N1CCC1C(N1CCC(OC)C(F)C1)=O 38144,Cc1ccnc2c(C(=O)NC(C)CCN(C)C(C34CC(C)(CCO3)C4)=O)cnn12 38145,c1(OC)ccc2cc(C(=O)NC3CCCN(C(=O)C(C)=CC4CC4)C3)sc2c1F 38146,c1(C(N(C2CCN(C(C3COCCO3)=O)CC2)CC)=O)cccnc1N 38147,c1(N2CCC(NC)CC2)ncnc(NCCC2CC(O)C2)c1C 38148,c1(CNC(=O)NCC(c2cccc(C)n2)CC)c(C)cc(C(=O)O)cc1C 38149,C(=O)(C1=NN2CCC(C)N=C2N1)N(C(C)CNC(=O)CCC1CC1)CC 38150,C1(C(=O)NCC(C2CC2)SC)CC2(CCN1C(=O)C=C1CCC(C)CC1)CC2 38151,C1(C(=O)NC(c2cc(OC)c(F)cc2)C)CC2OC(C)CC2N1 38152,C(CC(=O)N(CC)CC)(C(C)C)CC.n12nc(-c3ccc(F)cc3)nc1CCC2 38153,C1(NC(CNC2CC(C#N)C2)=O)CCn2nccc2C1 38154,N1(C(c2occ(C(=O)OC)c2)=O)CC2CC(NC(C3(N(C)C)CC3)=O)C1C2 38155,N1(C(C2CCCC(NC(c3ccc(C#N)cn3)=O)C2)=O)CCc2cncnc2C1 38156,C1(NC(C(C2CN(C(COCCN(C)C)=O)C2)O)=O)CCN(C)CC1(C)C 38157,Cc1nn(C)cc1CCNC(C1CN(C(=O)CC2(O)CCCC2)CC1C)=O 38158,N1(C(C(=Cc2ccc(C)cc2)C)=O)CC2(CC2)CC1CNC(=O)C1=CCCSC1 38159,C1(CCC)(NC(c2csnc2Cl)=O)CCN(C(c2cccc(O)n2)=O)CC1 38160,c1(-c2sc(C(N3CC(NC(C=C(C)C4CC4)=O)C3)=O)c(C)n2)c(C)nn(C)c1C 38161,c1(OC(CC)C)ccc(-c2nc(-c3cccnc3)nn2-c2ccnc(O)c2)cc1 38162,C1(C(N(CC(C)O)CCNC(=O)C(C2CC2)C2CC2)=O)CCc2nn[nH]c2C1 38163,c1(C(=O)NCC(CNC(CCN(C(CCC)C)C)=O)F)cc(O)cc(Cl)c1 38164,C1(C(=O)NCCN(C(C2(NC(=O)NCC)CCCC2)=O)C)COCCN1C 38165,C1(OC)(OC)COC(C(=O)NOc2ncccc2Br)C1.C1(O)CC1 38166,Cc1ccc(C(C)NC(C2CC=CCN2C(c2cnn(C)c2Cl)=O)=O)cc1 38167,c1(CN2C(CC)CN(C(c3cccc(C)c3)=O)CC2)ccc2nc(O)[nH]c2c1 38168,C1(C)(C(=O)NCC#CCNC(CCc2c(C)noc2Cl)=O)CCCCC1C 38169,C(C(=O)NCC1(F)CCC1)(C1CN(C(=O)CSC(C)(C)C)C1)OC 38170,c1(C(=O)NC2CCCC(N(C(CCC(=O)NC)=O)C)C2)oc2ccccc2c1C 38171,c1(C(=O)Nc2ccc(CC(=O)OCC)cc2)c(Br)cc(F)c(F)c1F 38172,CC(N=c1[nH]c(=NCCOCC2CCOCC2)[nH]c2c1COC2)c1ccn(C)n1 38173,CC1=NS(=O)(=O)NC=C1C(=O)NC1(CCCNC(C2(S(C)(=O)=O)CC2)=O)CC1 38174,C1(NC(c2c(C)noc2)=O)CC2CCC(C1C)N2c1ncccn1 38175,Cc1ccc2c(c1)CC(C(N1CC=CC(NC(=O)C(C)(Cl)Cl)C1)=O)S2(=O)=O 38176,C(=O)(CCCC(C)NC(=O)C(C1CCCCC1)F)NC(C(=O)OC)CO 38177,c1(C(=O)NCC2C3CN(C(C(C)n4cccc4)=O)C2C3)cc([N+](=O)[O-])ccc1Cl 38178,Cc1cn2c(C(=O)NCC3CCCCN3C(=O)CCC(N)=O)cnc2s1 38179,c1(CNC(=O)Nc2c(C)cncn2)ccnc2ccccc12 38180,Cc1ccc(OC(F)(F)F)c(C(=O)NC2CCC2NC(=O)C(C)n2cncn2)c1 38181,N(C1CCc2sc(Br)cc21)C(=O)OC(C)(C)C.c12cccc(c1)CNC(=O)N2 38182,C1(NC(=O)Nc2cncc(OCCO)c2)CCCCC1Nc1ncc(I)cn1 38183,C1(CC(=O)NCCCCC2C(C)C2)CCCN(C(c2nonc2N)=O)C1 38184,C1(C(=O)NC(C)(C)CCNC(=O)Cc2cnoc2)CC2(CCC2O)C1 38185,C1(O)(CNC(CC(=O)OC)=O)CCN(C(=O)C(C)Sc2ccccn2)C1 38186,C1(NC(CCC2(C#N)CCC2)=O)CN(C(C2CC(=O)CCO2)=O)CC(F)(F)C1 38187,C1(CNC(c2ccc(SC)s2)=O)CC2CN(C(=O)CCN3CCCCC3)CC12 38188,S(=O)(=O)(c1cnn2c1OCCC2)NC(Cc1cc(C)[nH]n1)=O 38189,CCC(CS(C)(=O)=O)NC(C1CC(NC(=O)OC(C)(C)C)C1)=O 38190,N1(C(C(c2ccc(Cl)cc2)C)=O)CC(C)(C)CC1CNC(C1CC1F)=O 38191,N1(C(CC2(C)CC2)=O)CC2CCN(C(c3ccc4occc4n3)=O)CC2C1 38192,C1(C(N(C(C)CCNC(C23CC(C#N)(C2)C3)=O)C)=O)CC(=O)C12CCC2 38193,N1(C(CCC#C)=O)C(C(=O)Nc2ncncc2I)CC2CCCCC12 38194,CC(C)(C)CCC(F)C(=O)N1CCCC(F)(CNC(=O)CCn2cncn2)C1 38195,C1(CC(=O)NC2C(C(N)=O)C2)CCCC1NC(c1cc[nH]c1)=O 38196,C12(NC(C3N(C)C(=O)CCC3)=O)CCCC1CN(C(=O)C(C)(C)c1ccns1)C2 38197,C1(NC(=O)NCCC(CC)C)CCCN(C(=O)OC(C)(C)C)C1c1cncn1C 38198,C1(C(N2CC3CC(C2)O3)=O)CC2CC2N1C(C1CCNC(=O)C1)=O 38199,C1(CN(C(c2c(CC)cc[nH]2)=O)C)CCC(NC(C2CC=CCC2C)=O)CC1 38200,N1(CCC)CCCC(C(N2CCC(N(C(=O)C(F)OC)C)CC2)=O)C1 38201,c1(C(=O)NC2CC(CNC(c3cc(F)c[nH]3)=O)C2)cnc2ccccn12 38202,c1(C(=O)NC2CC(CNC(CCc3cnn(C)n3)=O)C2)cccc(=O)o1 38203,c1(CNC(c2n(CCC)ncc2)=O)nnn(C)c1C(N1CC(N(C)C2CC2)C1)=O 38204,C1(C(N2C(C)(C(NOC(C=C)C)=O)C=CC2)=O)CC2CC(=O)C1C2 38205,C(=O)(C(CO)NC(=O)COC(F)F)NC1C(C(C)(F)F)C1 38206,c1(COC)cc(C(=O)NC(C(=O)NCC23CCCC2C3)c2ccco2)n[nH]1 38207,c1(C(=O)NCC(C)NC(=O)CC2CC=CCN2C)ccc2c(c1)CCC(C)(C)O2 38208,C1(C(=O)NCC=CC(=O)NCC2(CO)CCCCO2)(OC)CCOCC1 38209,CCCCC(CC)CC(=O)NCC(C)(C)C(=O)NCCS(C)(=O)=O 38210,Cc1cn2c(n1)C(C(=O)NC13CCC1CN(C(c1cc(=O)n(C)o1)=O)C3)CCC2 38211,Cn1nc(C(F)(F)F)c([N+](=O)[O-])c1N1C2CCC1C(C)C(NC(c1ccon1)=O)C2 38212,c1(C(=O)NC2C3(CN(C(C4CC(C)C4)=O)C3)CCC2)ccc2c(n1)OCC(=O)N2 38213,N1(CC(CCC)OC)CCCC(c2nn[nH]n2)(C(C)C)C1 38214,c1(C(N2CCN(C(CN3CCC(C)(O)C3)=O)CC2)=O)c(F)ccc(Br)c1F 38215,N1(C(c2snc(C)c2N)=O)CCCC(CC(=O)N(CC(C)(O)C2CC2)C)CC1 38216,C(=O)(CCCN=[N+]=[N-])N(CCOCCNC(C1(CC=C)COC1)=O)C 38217,C1(CNC(c2cc(C)oc2)=O)CN(C(=O)CSC(C)(C)C)CCC1C 38218,c1(CSC)cccc(C(=O)NCC(O)CN(C)C(C2CC(CF)C2)=O)c1 38219,c1(C(N(CCC2CCN(C(CC(C)F)=O)CC2)C)=O)ccn2cncc2c1 38220,C1(F)(CNC(CN(C)C(N)=O)=O)CCCN(C(=O)C(F)Cc2ccccc2)CC1 38221,CC(C)(CC(F)(F)F)C(=O)NCC1COCC1NC(=O)Cc1ccccc1 38222,CC1(C)CCCN(C(c2ccc(N)c(F)c2)=O)C1CNC(=O)C#CC1CCC1 38223,C1(NC(c2n(CC)ncc2Br)=O)CCCN(C(=O)CC2(OC)CCC2)CC1 38224,Cn1cc(C#CCNC(c2cc(CNC(C3CCCC(=O)N3)=O)cs2)=O)cn1 38225,CC1CCCCC1C(=O)NCC1CCN(c2nccc(C(F)(F)F)n2)C1 38226,c1(CNC(=O)COCCCF)ccc2c(c1)CN(C(c1cc(CO)ccn1)=O)C2 38227,C1(NC(C(CC=CC)C)=O)CCCOC12CCN(C(=O)Cc1cc(C)on1)CC2 38228,C1(C(=O)NCCCC2CCOC2)(COC)COc2ccccc2C1 38229,c1(CNc2c(C(=O)OC)cc(C)c(C)c2)ccc2c(c1)C(CCOC)C(=O)N2 38230,c1(CN(c2ncn(CCNC(CCOC)=O)c2)C(C)=O)ncccc1C#N 38231,CC1CN(C(=O)CCSCc2ccccn2)CCC1NC(=O)C=Cc1cc[nH]c1 38232,c1(-c2n(C(C)C3CC3)nc(CC3(C)CC3)n2)cc2ccncc2s1 38233,c1(C(N2CCCC(CNC(Cc3nc(C)oc3)=O)C2)=O)cc(S(N)(=O)=O)cnc1C 38234,C1(C(=O)NOCCO)(CC=C)CCCN1C(C1CCC(F)CC1)=O 38235,c1(C(N(CCC(C(C)C)NC(=O)CS(C)(=O)=O)C)=O)ccc2c(n1)CCO2 38236,CCC(CC)CC(F)C(=O)N1CCC2CCCC12C(=O)NC(C)C1CC1 38237,c1(C(=O)NCCCCCN(C(C=CCOC)=O)C)c(OC(C)C)ccnc1F 38238,N1(C(C(C=C)CC)=O)CCOC2(CCN(C(=O)Cc3ccco3)C2)C1 38239,C(=O)(C(F)(CNC(=O)C(C#N)C(C)C)C(C)C)N1CCC(OCC#C)C1 38240,C(=O)(C(O)C(O)c1ccccc1)N(CCCCNC(C(=O)N(C)C)=O)C 38241,N1(C(C(c2ccc(F)cc2)C)=O)CCC(C(=O)NCc2occc2C(=O)O)CC1 38242,C1(C(N2CCC3CC23)=O)COCCC1NC(C12CCN(CC1)C2)=O 38243,CCC(O)C(C)C(=O)N1CCN(C(C2CCCC2C(=O)OC)=O)CC1C1CC1 38244,c1(C(N2C(C)(CNC(=O)C=CC3CC3)CCC2)=O)occ2c1CCOC2 38245,c1(NC(C2C(C(N3CC4C(C(=O)OC)(C4)C3)=O)C2)=O)cncc(F)c1I 38246,c1(CC)cccnc1C(=O)NCC(C)N(C)C(c1ccc(-c2cccs2)[nH]1)=O 38247,C=C(C)C1OCCC1CNC(=O)NC(c1cccc(Br)n1)C 38248,CCC(C(C)(C)O)NC(=O)CC1CCN(C(=O)C(c2ccnn2C)C)CC1 38249,c1(C(=O)NC2CN(C(C(c3cnccn3)C)=O)CC2O)nsc2ccccc12 38250,c1(SC)cc(C(N2CC3CC2CN3C(c2cn[nH]c2)=O)=O)cc(SC)c1 38251,C1(C(N(Cc2n(CC)ncc2)CC)=O)CN(C(c2cc(OC)no2)=O)CC1OC 38252,C1(C(=O)NC(C2CN(C(C(CC#C)(C)C)=O)C2)C)CC2(C1)CC1(CC1)C2 38253,c1(NC(CNCC(CC(=O)NCC(=O)NCC(C)C)C)=O)coc2ccccc12 38254,c1(CN2CCC(C)(C(=O)NCCC)C2)cc2ccccc2s1 38255,N1(C(CC=C)=O)CC2CCC(NC(C3CCN(C(C)C)CC3)=O)CC2C1 38256,c1(CNC(CCCNC(N)=O)=O)cncc(C(=O)NC2COC(C(F)F)C2)c1 38257,c1(C(C)=O)cccc(CC(=O)NCCC2CCN(C(=O)C=C3CCC(C)C3)C2)c1 38258,C(=O)(CCCNC(C)=O)NCC(COC)NC(=O)C(CC1CCC1)OC 38259,c1(NC2CC3CC(CO)CC23)nc(CC2(c3cn(C)nc3)CC2)c2ccsc2n1 38260,C(=O)(CC(C)C(C)C(C)C)N(C)CC1(O)CN(C(c2cc(C)nc(C)c2)=O)C1 38261,C1(CNC(C(C)OC)=O)CN(C(c2cc(C)c(Cl)cc2F)=O)CCC1(C)C 38262,N1(C(=O)COCCF)CCC2CN(C(=O)CSCc3ccc(Cl)cc3)C2C1 38263,C12CCN(CC1)CC1C(CCCC1)S2.c1(OC(F)(F)F)nnc(Br)s1 38264,N1(C(C(C)(C)C#N)=O)CCC(F)(F)C(CNC(C2(C)CNC(=O)C2)=O)C1 38265,N1(C(C2CCCC(CF)C2)=O)CCOC2(CCC(NC(C3CC(O)C3)=O)CC2)C1 38266,c1(C(=O)NCC2N(C(CC(=O)OC)=O)CCN(C)C2)ccccc1N=S(C)(C)=O 38267,C1(C(N(C2CCN(C(C3(C)CCC(C)CC3)=O)C2)CC)=O)CCc2nn[nH]c2C1 38268,CC(CC(=O)NC(C)(C)CCN(C(=O)CC(C)n1ccnc1)C)c1ccccc1 38269,C(C(=O)NCCCCC(C)NC(c1cnc(C2CCC2)o1)=O)(C(C)C)SCC 38270,c1(C(N2C(C(C(=O)NC3CC4(CN(C)C4)C3)(C)C)CCC2)=O)ccn2cncc2c1 38271,c1(OCC)cc(NC(c2ccc(-c3cn[nH]c3)cc2)C)cc(Br)c1 38272,C12(C(=O)NCC(CC)NC(C3COC(=O)N3C)=O)CC(CO)(C1)OC2(C)C 38273,C1(C(=O)NCC2(COC)CCCN2C(=O)CN=S(C)(C)=O)COC2(CCC2)C1 38274,c1(C(N(CCNC(C(CC)CC(F)F)=O)C2CC2)=O)ccc2c(c1)CCCC2=O 38275,c1(CC)c(C(=O)NCC2(NC(=O)Cn3ccnc3C)CCOC2)cnn1C 38276,N1(C(COC(C)(C)C)=O)CC2=C(C1)CN(C(c1ccc(C3CCOC3)s1)=O)C2 38277,CC1CCN(C(c2cnc(O)o2)=O)CC1CC(=O)NCCC1CCCC12CC2 38278,C(=O)(C1CCc2cccc(=O)n21)NC1C(OC)CN(C(C2(C(=O)OC)CC2)=O)C1 38279,C(=O)(C(F)CC(C)(C)C)NCc1ccc(C(=O)NCC2(OC)CCCC2)nc1 38280,c1(C(=O)OC(C)(C)C)cccc(CN(C)C)n1.C12(C)CCN1C2=O 38281,C(=O)(C(C(C)(C)C)OC(C)(C)C)N(C)CC1(N(C)C)CCC1.C12CCN(C1)C2=O 38282,N1(CC)C(=O)CCC1C(=O)NC(C1CCCC1)CNC(=O)C(=C1CCCCC1)F 38283,C(C1CCN(C(C2(C)CC(F)C2)=O)CC1)=CC(=O)NC1(CC=C)CC1 38284,N1(C(C=CC2(C)COC2)=O)CC2(CCN(C(c3ccccc3C(F)(F)F)=O)C2)C1 38285,c1(C(=O)NC(C)C(CO)NC(c2cc3n(c2)CCSC3)=O)cccn2nccc12 38286,C1(CNC(CCCc2ncc(C)o2)=O)CC(NC(=O)CNC=O)C12CCC2 38287,Cn1cc(C(=O)NCCCNC(=O)C(F)CC2CCCCC2)ncc1=O 38288,CCC(C)CCCCC(=O)NCC(C)N(C(c1ccc(OCCF)cn1)=O)CC 38289,C1(NCc2ncc(C(C)(C)C)s2)COC2CCCCC12 38290,Cc1cc(C(=O)NCC2(NC(=O)C=Cc3ccc(=N)[nH]c3)CC2)c2c(c1)CCC2 38291,Cc1cc(F)ccc1NC(N1CCC(C)(NC(=O)C(=O)NCC(F)F)CC1)=O 38292,Cc1ccnc(O)c1C(=O)NC(CNC(c1ccnn1CC(F)F)=O)C1CC1 38293,C(=O)(C(CC)(CC)CC)N1C(C)(CC(=O)NC(C(=O)OCC)CO)CC1 38294,C1(NC(=O)C(F)C2CCC2)CN(C(=O)CN2CCCCC2=O)CC12CC2 38295,N1(C(C=CC)=O)CCN(C(=O)C(C)N(C)C(C)=O)C2(CC2)C1 38296,c1(C(N(CCCNC(C2CCCNS2(=O)=O)=O)CC)=O)ccc(Cl)c(OC)c1N 38297,C1(C(=O)NCCC(C)NC(c2cccc(-n3cccc3)n2)=O)CC=CCC1C 38298,C12=NC(=NCC3CN(CC3C(F)(F)F)C1=O)NC=C2Cl.c1(OCC)ccoc1 38299,CCC(C(=O)NCC(C)CNC(=O)Cc1cccc(OC)c1F)C(F)(F)F 38300,C1(C(F)(F)F)(OC)CCCN(CC2CCC(C#N)CC2)C1 38301,CC1(C)CC(CNC(C2CC3(CCCO3)C2)=O)CN1C(c1ccc(C2CC2)o1)=O 38302,CCCCCS(=O)(=O)CC(=O)N1CC2CC2(NC(c2cc(F)c(N)c(F)c2)=O)C1 38303,CCC(C(=O)NC(CO)C(=O)NCCCCO)n1ccnc1 38304,Cc1cc(O)c(C(N2CCCC(C(C)NC(=O)Cn3nccc3C)C2)=O)cc1F 38305,c1(C(N(C(C)CNC(=O)CC2CC(F)C2)C)=O)c[nH]nc1Cl 38306,C1(NC(C(=O)N(C)C)=O)CC(F)CN(C(=O)Cn2cccc(N)c2=O)C1 38307,C#CCC(C)(C(=O)NC(CC1CC1)CO)NC(c1ncn(C(C)C)n1)=O 38308,N1(C(C(C)(C)OC)=O)CC2(CCC2)CC1CNC(=O)C#CC1CCCO1 38309,C1(NC(CC2N(C)CC=CC2)=O)CCN(C(=O)CC2CN3CCC2CC3)CC1O 38310,c1(C(=O)NCCOC2CN(C(c3nn(CC)c(C)c3)=O)C2)sc(C)c(C)c1C 38311,c1(C(=O)NC2(C)CN(C(C3(C)CCCS3(=O)=O)=O)C2)ccc(F)c(C(F)F)c1 38312,C=CC1OCCC1C(N1CCC(CCN(C(=O)CC(O)CN(C)C)C)CC1)=O 38313,N1(C(C2C(C3C(C)C3)C2)=O)CCC(O)(CN(C)C(c2cn3ccsc3n2)=O)CC1 38314,C12(NC(CC3(NC(C)=O)CC3)=O)CCCC1CN(C(=O)Cc1c(C)cccc1Cl)C2 38315,c1(C(=O)NCCC(C)N(C(=O)C(O)CC[S+](C)C)C)nnc(O)c2ccccc12 38316,c1(C(=O)NC(C(=O)NC(CC)CCCO)c2ccoc2)c[nH]c(C)cc1=O 38317,Cc1cc(F)sc1C(=O)NC1CCCC1CNC(c1cnc(O)o1)=O 38318,N1(C(C2(CC=C)CCC2)=O)CC2CC1CN2C(C1CC1(F)Cl)=O 38319,N1(C(C(OC)OC)=O)C2CCC1CC(NC(C1CCNC(=O)C1)=O)C2 38320,CC1CCN(C(=O)CC2CCC2(F)F)CCN1C(c1noc2c1CCCC2)=O 38321,n1(C2CCN(C(C(=O)N(c3c(C)ncn3C)C(C)C)=O)CC2)c(C)nc2cnccc12 38322,Cc1ccc(C(=O)NC2(C)CC(NC(C3(C)COC3)=O)C2)c(C)c1Br 38323,c1(CNC(=O)CN(C(=O)COc2ccsn2)C2CCC2)ccc(O)nc1 38324,Cc1oc2ccccc2c1C(N1CCN(C(=O)CC2COC(C)(C)C2)C(C)C1)=O 38325,C1(C(N2CCC(O)(Cn3cc(C4CCCC4O)nn3)C2)=O)CCCC2(CCC2)O1 38326,N1(C(C23CCC(C(=O)OC)(C2)C3)=O)CCC2CCCN(C(C3(C)CCC3)=O)C2C1 38327,N1(C(C2(C3(C)CC3)CC2)=O)CCOCC(C(=O)NCCN2CCC3CC23)C1 38328,C(=O)(C(F)C(=O)N(C)CC1CCCCN1C(=O)C(C)(C)OCC(F)(F)F)OCC 38329,CCCC(C)(CCC)C(=O)NC1CC(NC(=O)CN(C)CCOC)CC1O 38330,C1(CCC)(NC(=O)C(C)n2cccn2)CCCN(C(c2cn3c(n2)SCC3)=O)C1 38331,c1(C(=O)NCC2CC(NC(c3nc(OC)oc3)=O)C2(C)C)ccc2c(c1)OCO2 38332,c1(CC(=O)NCC2(NC(C(CSC)O)=O)CCOC2)ccc(Cl)cc1C 38333,N1(C(c2cncc(N)c2)=O)CC2CCC1C1CN(C(c3cnc(O)o3)=O)CC21 38334,c1(C(CC)C(=O)N(CCCN2CCCC2)C)ccc2c(c1)OCO2 38335,Cc1conc1C(=O)NC(C1CN(C(c2cnn(C(C)C)n2)=O)C1)C 38336,C1(C(=O)NCC2(C(C)(C)O)CN(C(CSCC=C)=O)C2)CCCCCC1(F)F 38337,CC(C(C)(C)C(=O)NCC1(CC2CC2)CC1)NC(c1cnc(CO)o1)=O 38338,C1(C(=O)NCc2c(CC)cncc2)CCCN1NC(=O)C(F)C(F)(F)F 38339,C1(C)(C(=O)NC)CCCN1C(c1cn(CCNC(=O)CC2(C#N)CC2)cn1)=O 38340,C(C(F)(F)C(F)(F)F)OCC1C(N(CC(=O)NC(=O)CC)CCC)CC1 38341,C=CC(C)(CC)C(=O)N1CC(CNC(C2(c3ccccc3)CC2C(F)(F)F)=O)C1 38342,n1(CCOC)ccc2cc(NC(c3cccc4c3COC4)=O)ccc12 38343,c1(CC)cccnc1C(=O)NC1CC(C)N(C(=O)CC(C)n2ccnc2)C1 38344,Cc1cc(NC(C2CC3CC3N2S(=O)(=O)c2cn[nH]c2)=O)c(C)cc1Br 38345,n1(CCCSCC)nnnc1C(c1ccn(C(C)C)c1)NCc1noc(C)n1 38346,C1(C(=O)NC(C2(C(N3CCCC(CC(C)C)C3)=O)CC2)C)CC(C2CC2)=NO1 38347,c1(CN(CC(C(C)C)O)C=O)nc(Br)sc1Br 38348,c1(C(=O)NCC(CC)NC(C2(C3CC3)CCCO2)=O)[nH]c2ccc(C)cc2c1C 38349,C#CCC(O)C(=O)N(CCC(C)NC(c1cc(COC)oc1C)=O)C 38350,C1(CC(=O)NCCN(C2CCCCCC2)C(=O)C=C2CCC2)CCS(=O)(=O)C1 38351,C1(OC)CN(C(=O)Cn2nnc(C(C)(C)C)n2)CC1NC(=O)CS(=O)(=O)N(C)C 38352,N1(C(c2c(C)csc2)=O)CCCCC1CNC(c1ccc(-c2ccco2)s1)=O 38353,N1(C(C(C)Cc2ccnn2C)=O)CC(CNC(=O)C(C)C(F)(F)F)C(F)(F)C1 38354,Cc1n[nH]cc1C(C(=O)NC(C)C)N(C)CCC1CCCCC1 38355,C1(C(=O)NC(CC=C)COC)(C(=O)OCC)CCCNC1 38356,C1(CNC(C(=O)N(C)Cc2ccn(CC)n2)=O)C2CCCCCC12 38357,N1(C(CN(CCC#C)C)=O)CC2CC(C1)CN(C(=O)CC1CC(OC)C1)C2 38358,C1(NC(c2c(Cl)cn(CC)n2)=O)CC2CC(C1)CN(C(C1CC3C=CC1O3)=O)C2 38359,N1(C(C)=O)CCN(S(=O)(=O)N(C)CC2Cc3nccn3C2)CC1 38360,C1(C(=O)NCC(CN(C)C(C2(C(F)F)CC2)=O)O)CCC=CCCC1 38361,C1(COC)C(O)C(O)CCN1C(C1CCCN(c2ccnn2C)C1)=O 38362,CC1(C)CC(C#N)(CNC(=O)COC2CN(C(=O)CC3CCCCC3F)C2)C1 38363,c1(C(C)=O)ccc(F)cc1NC(C1CC(CN2CCCC2)C1)=O 38364,Cc1cc(C)c(C(=O)NC2CCC(F)(CNC(c3cccn3C(C)C)=O)C2)cn1 38365,c1(C(=O)NCC(C=C)O)nc(CNC(=O)CN(C)C(C)=O)oc1C 38366,c1(C(N2CC(OC)C(NC(=O)C(CO)NC(N)=O)C2)=O)c(C)oc(C)c1Br 38367,c1(C(=O)NCCCCNC(c2c(SC)cccc2F)=O)ncnc2ccsc12 38368,n1(CC(N2CC(C(C)NC(c3n(C=C)nnc3)=O)C2)=O)nnc2ccccc12 38369,C(CCCCC(=O)N1CC=CC1C(=O)NCCN1CCCCCC1)=CC 38370,CCCC(C(=O)N1CCCC(N(C(=O)C(C)OCC(C)C)CC)C1)N(C)C 38371,CC1(C)CC(C(F)(F)F)(C(=O)NCC2CCC2NC(=O)CSc2ccccn2)C1 38372,N#Cc1n[nH]c(=NC2CCCC23CN(C(c2c[nH]cc(Cl)c2=O)=O)C3)s1 38373,CC1CC=C(C(=O)N2CCCCC(NC(C3NC(=O)OC3C)=O)C2)CC1 38374,C1(C(N2CCC(OC)C2C(C)C)=O)COC2(C1)CN(C(c1cccc(C)n1)=O)C2 38375,C(=O)(C(C)CCCC(C)C)NC(CNC(C(=Cc1cn[nH]c1)C)=O)CO 38376,N1(C(C2COC(=O)O2)=O)CC23CCCC2(C1)CN(C(c1cnc(O)s1)=O)C3 38377,CC1CN(C(=O)C(c2ccc(F)cc2)F)C(C)CN1C(=O)C1=CCSC1 38378,N(C1COc2c(Cl)cccc21)C(N(C)Cc1ccccc1I)=O 38379,C12(NC(C3(C#N)CC(C)C3)=O)CCCC1N(C(=O)CCOCC(F)(F)F)CCC2 38380,c1(C(=O)Nc2cc(C)cc(O)c2)cn(C)c2ccc(-c3cccc(F)c3C)cc12 38381,CC1CN2CCN1C(C(N1CC3(CC(NC(c4cc[nH]c4)=O)C3)C1)=O)C2 38382,CC1(C)CCN(C(=O)C=C2CCC2)CC1C(=O)NCC1CC(O)C(O)C1 38383,C1(CCNC(CC2C(C)CCC2)=O)CCCN(C(=O)CC(C)(C)O)CC1 38384,C1(C(C)(C)O)(CNC(=O)CNC2CCCC2)CN(C(=O)CC2CCCC2)C1 38385,N1(CC)C(=O)CCC1CC(=O)NCCN(C(C1COCC1(C)C)=O)CC1CC1 38386,C1(N(CC(=O)Nc2onc(C)n2)C)CCCN(c2ccccc2)C1=O 38387,N1(C(c2sc(C(F)(F)F)nc2Br)=O)CCS(=O)C(F)(F)C1 38388,c1(NC(C2CN(C(C3CNC(=O)O3)=O)CC(F)C2)=O)nc(Cl)c(Cl)nc1CO 38389,C(C(C)C(F)C(=O)NCC1C(C)(C)C1(C)C)NC(c1noc(CC)c1C)=O 38390,C1(COC)(NC(=O)C(c2ccccc2)F)CCN(C(=O)CCOC(C)=O)CC1 38391,C(=O)(NNC(=O)C(CN)CC(C)C)c1nc(C)c(I)cc1 38392,N1(C(C(CC(C)(C)C)NC(c2cnn(CC)c2C)=O)=O)CC(C)C12CCOCC2 38393,Cc1nc(C(C(=O)NC2(C)CC2)N(C)C(c2ccc(F)cc2)C)sc1C 38394,c1(CCNC(C(C2CCN(C(c3ccn(C)n3)=O)C2)(C)C)=O)ccc(F)cc1 38395,CC1CN(C)CC(C(N2CCCN(C(=O)CN3C(=O)CNC3=O)CC2)=O)O1 38396,C1(OC)CC(CNC(=O)CC2(O)CC2)N(C(=O)CCn2cccn2)C1 38397,c1(C(N(CCN(C(CCc2cnc(C)s2)=O)C(C)C)C)=O)ccccc1N(C)C 38398,C1(COC(N2CC(NC(N(C)C)=O)C2)=O)(CCl)CCSCC1.C(C)(C)C 38399,c1(C(=O)NCC2(O)CN(C(C3CC3(C)C(F)(F)F)=O)C2)ccccc1C1CCC1 38400,C(=O)(C(C)C(O)CC)NCC1(C(=O)NC2(CC=C)CCCCC2)CCCC1 38401,c1(CC(=O)NCC2CCN(C(=O)CCCc3ccsc3)CC2)ccc(O)c(Cl)c1 38402,C(C1=CCN(C(c2ccsc2)=O)CC1)NC(c1cn(C2CCC2O)nn1)=O 38403,C1(C(N2CCN(C(c3n(C)nnc3)=O)CC2CCO)=O)CC2CCCCCC12 38404,C1(NC(c2cc(CCC)ncc2)=O)CCN(C(c2sccc2F)=O)CC1C(N)=O 38405,CC1(C)CC(=O)N(CC(=O)NC2C=CCN(C(c3cccc(F)n3)=O)C2)C1=O 38406,c1(C(=O)OC)cccc(NC(=O)NCc2ccncc2C(C)C)c1OC 38407,C=CC1CN(C(=O)C(c2cscc2Br)=O)CC1NC(=O)C(C(C)C)OC 38408,C1(C(=O)NC(CCCCNC(c2cc(C(C)C)n(C)n2)=O)C)CC2CCC(C1)S2 38409,c1(C(N(C2CCCCC2NC(C2(C)COC2)=O)C)=O)ccc2c(c1)OC(C)(C)C2 38410,N1(C(c2cncc(N)c2)=O)CC2CCC2(CCNC(=O)C(=C2CCCCC2)F)C1 38411,c1(CC)ccc(NC(C2CCN2C(c2cc(OC)cc(Cl)c2)=O)=O)c(O)c1 38412,C1(NC(c2c(CC)cco2)=O)CCN(C(C2(C)CCCN2C)=O)CC1O 38413,Cc1c(NCC2(CCO)CC2)ncnc1N1CCN(c2ncccn2)CC1 38414,C1(C)(C(N(CCCNC(c2c(C(=O)OC)cco2)=O)C)=O)CCOC1C 38415,c1(C(=O)NC2CC(C(N(C3CC3)CC)=O)C2(C)C)cc(C)c(C)nn1 38416,C1(NC(c2ccc(CCO)cc2)=O)CN(C(=O)C2=CCC2)C2(CCOCC2)C1 38417,C1(NC(C(CC=C)CNC(=O)C=C(C)C(F)F)=O)CC2CC1CC21CC1 38418,C1(C(N2CCCN(C(c3ccc4cc[nH]c4n3)=O)CC2)=O)CCc2n[nH]cc2C1 38419,N1(C(CC2(CC(=O)OC)CC2)=O)CCC(C)(CNC(=O)COC2CC=CC2)C1 38420,c1(C(N2CCC(N(C(c3ncc[nH]c3=O)=O)CC)C2)=O)cc2c(ccn2C)[nH]1 38421,C1(CC(=O)Nc2ccc(Cl)cc2)CCN(S(=O)(=O)CC2CC2CC(=O)O)C1(C)C 38422,c1(C(=O)NCCN(C(=O)Cc2cc(Cl)ccc2O)CC)cnc2ncccc2c1 38423,C1(N(C(=O)COC(C)(C)CC)CC)CCN(C(c2nonc2N)=O)CC1 38424,N1(C(c2c(CC)nns2)=O)CCN(C(=O)Cc2ccc(C)c(C)c2)CC1C(C)C 38425,N1(C(C(CC)=CC)=O)CCC(CNC(=O)CCc2ccc(OC)c(Cl)c2)C(C)C1 38426,c1(C(N2CC(C)(C(=O)Nc3cncc(C(C)(C)C)c3)C2)=O)ccc(Br)nc1Br 38427,c1(C(N2CCCC(N(C)Cc3cc(C)no3)C2)=O)n[nH]c(C)c1[N+](=O)[O-] 38428,c1(C(N2C3CC(NC(c4n(CC)nnc4)=O)C2CC3)=O)cccc2c1OCCO2 38429,N1(C(c2ncn(CC)c2)=O)C2CCC1CC(CNC(=O)C(=Cc1cscn1)F)C2 38430,CCCCCCCCC(C)CC(=O)NC1CC(CNC(=O)C(F)(F)C(F)(F)F)C1 38431,C1(C(=O)OC)CN(C(=O)NCC2CC(C)(C)OC2(C)C)C2CCCC2O1 38432,N1(C(c2c(C)nc(N(C)C)s2)=O)CCCC12CCCN(C(=O)C(O)C1CC1)C2 38433,c1(OC)ccc(OC)c(C(N2CCC(C)(CNC(C3(C)CC(C)(C)C3)=O)C2)=O)n1 38434,Cc1ccc(C2CC2C)cc1Br.N1(N(C)Cn2cc(CCO)nn2)CCOCC1 38435,c1(C(=O)NCCN(C(=O)C(O)CC(F)F)C)cccc(S(=O)(=O)C2CC2)c1 38436,O(NC(=O)CC(CCCC)NC(=O)C(CO)C(F)(F)F)CCC(=C)C 38437,C1(CNC(c2nc(CCC)sc2)=O)C(O)C(O)CN1C(C1CCCCS1(=O)=O)=O 38438,C1(C(=O)Nc2cn3c(n2)CCC3)CCN(C(=O)COc2cccnc2)CC1F 38439,c1(C(C(=O)NC(C(C)NC(=O)CO)C)F)cccc(F)c1Cl 38440,C1(c2cccs2)(C(=O)NC(C#C)(C)C)CCN(C)C1 38441,C(=O)(CC(C1CC1)C1CC1)NC(CN(C(C(=O)NCC)=O)C)CC 38442,CC1(CNC(c2cocn2)=O)COCCN(C(c2scnc2-c2cccs2)=O)C1 38443,Cc1cccc(C)c1CC(=O)NC1CC2(C1)CC(NC(C1(F)C3CCCC13)=O)C2 38444,c1(NC(C2(O)CCN(C(c3cnc(Cl)c(Br)c3)=O)C2)=O)cnc2n[nH]c(Br)c2c1 38445,N1(C(COCCC#C)=O)CC2CCC2(CC(=O)NC(C)COC)C1 38446,c1(N2CC(C)S(=O)CC2)ncc(S(=O)(=O)NCCC2(CO)CCC2)cc1Cl 38447,Cc1c(C(=O)NC2CC3CCC2N3c2cc(OC3CC3)ncn2)cncc1Cl 38448,C=CCC(CC(=O)NCc1ncoc1C1CC1)NC(=O)C(CCC)N(C)C 38449,C1(N(C(c2cccc(Br)c2)=O)CC)CN(C(=O)CN2CCC2C)C(C)(C)C1 38450,c1(C(C)NC2(C)CCC(=O)NC2=O)cccc(S(=O)(=O)C(=O)N(C)C)c1 38451,c1(C(N2CCN(C(C(C(CC)C)C)=O)C(C(C)C)C2)=O)cc(C)c2[nH]nnc2c1 38452,c1(C(=O)NCCN(C(C2(N(C)CC)CC2)=O)C)c(Cl)nc2sc(C)cn12 38453,C1(C(C)NC(CC=C)=O)CCCCN1C(c1nc(C(F)(F)F)sc1C)=O 38454,N1(C(C2C3CN(C(CC4(C)CCCC4O)=O)CC32)=O)CCn2cncc2C1 38455,c1(C(=O)NC2CC3(CC(NC(CCC(CC)C)=O)C3)C2)ccc2c(c1)CCN2 38456,C1(NC(C2CC(CC)OCC2)=O)CC2CCC1CN2C(c1cc[nH]c1C1CC1)=O 38457,C1(CC(=O)NCC2CC3(CCC3)CO2)C2CCCC2N1C(=O)C1=CCCC1 38458,C1(NC(CCCC=C)=O)CCC2(CC1)CC2NC(c1c(SC)cnn1C)=O 38459,n1(CC(=O)NC(C2CCN(C(C3CN(C4CCOC4)C3)=O)C2)C)cc(Cl)cn1 38460,C1(C(=O)NCCOCCC#C)CC(O)CN1C(C1(CC=C)COC1)=O 38461,C=C(C)CCC(C)NC(=O)C(O)CNC(c1cncc(OC)c1)=O 38462,CC1COC(C(=O)NCc2csc(CNC(C3OCCO3)=O)n2)C1 38463,CCN=c1ccc(C(=O)NCC2(F)CCC(CNC(=O)CC3CC3)C2)c[nH]1 38464,c1(C(=O)NCCCn2cc(C(C)(C)C)nn2)ccc(CO)cc1F 38465,c1(C(N2CCC(CNC(C(C=C)O)=O)CC2C)=O)c[nH]c2c(F)cccc12 38466,O=S(=O)(CCCCC1CC1)NC1(c2ccc(F)cc2)CCCCC1 38467,N1(C(Cc2ncc(C)s2)=O)CC2CC(NC(c3cn(C)nc3C(F)(F)F)=O)C2C1 38468,CC1=C(C(=O)N2CCC(C)(NC(C3CC4CC4C3)=O)C2)CCCO1 38469,c1(C(=O)NC(C2CCOCC2)(C)C)ccc(CNC(C2CC3(CC3)CO2)=O)cn1 38470,c1(CC)oc(C(=O)NCCC2(O)CN(C(=O)CCC(C)OC)C2)cc1C(=O)OC 38471,c1(C(=O)NC2(CCOC)CCN(C(c3cnncc3O)=O)C2)c[nH]cc(C)c1=O 38472,Cc1cc(F)ccc1-n1cc(O)c(C(=O)OCC2C=CCC2)n1 38473,c1(NC(C2CN(C(c3c(I)ccnc3Cl)=O)CCN2)=O)ccc(Br)cc1Cl 38474,CC1CCC(C)(C(=O)NC2CCCC2NC(=O)CCC2OCCO2)C1(C)C 38475,c1(CNC(C2CCC3(CN(C(C(C)=O)=O)C3)O2)=O)ccc2ncccc2c1 38476,c1(C(N2CCC(CNC(C3(C#N)CCCO3)=O)C2)=O)cn2cc(Cl)cnc2n1 38477,C1(CC(N2CC(CC(C)NC(=O)Cc3cnsc3)C2)=O)OCCC1(C)C 38478,C12(C(N(C3CCCN(C(C(CC#C)O)=O)C3)CCO)=O)CCOC(C)(C1)C2 38479,CN=c1[nH]cc(C(=O)NC2CCOCC2C(=O)NCc2cc(Cl)ccn2)s1 38480,C12(NC(c3[nH]c4cc(C)sc4c3)=O)CCCCC1N(C(=O)Cn1cnnn1)CC2 38481,N1(C(=O)NC(c2nc(C(=O)OCC)c(N)s2)C)CC(C2CCC2)CCC1C 38482,C(=O)(CC(O)(c1ccccc1)C1CC1)NCC(C)NC(c1c[nH]c(Br)c1)=O 38483,c1(C(=O)NCC2CC3CCC2N3C(=O)CCSC(F)(F)F)coc2c1CCCC2 38484,C1(C(N2C(CNC(C3CC4(CCC4)C3)=O)CC3CC32)=O)CCc2nc(O)[nH]c2C1 38485,C1(C(=O)NCC(CCNC(c2ccc(Cl)o2)=O)OC)CCCCC12CC2 38486,c1(C(=O)NC2CC(CNC(C3CC4CC4C3)=O)C2)cccc2ccnn12 38487,N1(CC(=O)N(CC(C)NC(=O)C(O)C(F)F)CC)C(=O)Cc2ccccc2C1=O 38488,N1(C(c2nn(C)c(=O)cc2)=O)CCC(NC(=O)CC2CC2C(F)(F)F)CC(C)(C)C1 38489,N1(C(C=CC(C)(C)C)=O)CC2CC1CN2C(c1[nH]ccc1-c1ccccc1)=O 38490,c1(C(=O)NC2(C)CCC(NC(=O)C(N)=O)CC2)coc(C#Cc2ccccc2)c1 38491,c1(OC(C)C)cnc(=NCCC(C)NC(C2CCc3nn[nH]c3C2)=O)[nH]c1 38492,O=C(CC(C(F)F)c1ccccc1F)NCC=CCNC(C1CC=CCC1)=O 38493,N1(C(c2cc(OC)ncc2F)=O)CCCN(C(C2CC3CCC(C2)O3)=O)CC1C 38494,C1(C(N2C(Cc3c(C)cccc3)CCC2)=O)C2CC3C1C3C2F 38495,N1(C(CCC(=C)Cl)=O)CCCCC(CNC(c2ccn(C(F)F)n2)=O)CC1 38496,C(C(C)CC(=O)N(C(C)CN(C(=O)Cn1nc(C(F)(F)F)cc1C)C)C)OC 38497,C1(N(C)C(c2ncoc2Br)=O)CCC(NC(=O)CN2CC=CC2)CC1 38498,C(=O)(CC(O)CNC(=O)CCc1ccsc1)N(C(C1CCCC1)CO)C 38499,C(CC(=O)NCC1(C)CCN(C)C1)(C(F)(F)F)NC(C1(OC)CCOC1)=O 38500,C1(NC(CNC(C(C)(C)C)=O)=O)CN(C(=O)Cn2nnc(=O)[nH]2)CC12CC2 38501,CCCC(C)(O)CC(=O)NCC1(C)CN(C(c2nc(C)c(C)s2)=O)CC1C 38502,N1(C(C(C)C2CCCC2)=O)CCOC(C)(CNC(c2cc(CF)on2)=O)C1 38503,C1(C(=O)NC2C(c3cn(C)nc3)C2)N(C(=O)CC2CCC=CCC2)CCC1(C)C 38504,C(=O)(C(CC(C)CCC=C(C)C)N1CCC(C)(C)C1C)NCCSC 38505,Cc1ccc(CN2CCC(C(=O)NCc3cccnc3F)C(O)C2)cc1C#N 38506,CC(CN(C)C)N=c1[nH]c(N2CCC(C(C)(C)C)C2)nc2c(F)cccc12 38507,Cc1nc(O)ccc1C(N1C2CCC1C(CNC(C1CC3CCCC13)=O)C2)=O 38508,C(CNC(c1cc(Br)no1)=O)(C(C)(C)C)NC(c1ccc(C(=O)OC)s1)=O 38509,N1(C(c2cnc(-c3ccccc3)o2)C(=O)NCC=C)CC(=O)N2CCCCC2C1 38510,C(=O)(CCCC(C)C)NC1C(SC)CN(C(=O)C(C)Cc2ccco2)C1 38511,C=C(C)CC(C(=O)NC(C)C(=O)N(CC(C)O)CC1CC1)OC 38512,C1(CNC(c2n[nH]c(C)c2O)=O)(NC(=O)C(C)SC(F)(F)F)CCC(C)(C)CC1 38513,CC(=O)CCCC(=O)N1C2CCC(C2)C1C(=O)Nc1cn(C)nc1Cl 38514,c1(OC)ccc2oc(C(=O)NC3(C#N)CCN(Cc4ccccc4I)C3)cc2c1 38515,C1(N(C(C(CC)O)=O)C)C2CN(C(=O)CCCNC(=O)OC)CC12 38516,c1(OC)cc(CC(=O)NC(C)C(C)NC(=O)Cc2cccc(C)c2Cl)ccc1F 38517,c1(C(=O)NC2C(CNC(CSCC(C)C)=O)CCC2)nnc(O)cc1O 38518,Cc1cc(=O)n(C)cc1NC(C1CC12CC(NC(=O)C(C)CN(C)C)C2)=O 38519,C(=O)(C(C)C(O)C(C)C)NCCCC(C(N1CCCC(C)(CC)C1)=O)O 38520,C1(NC(C2CCCN2C(c2cc(-c3ccccn3)[nH]n2)=O)=O)C2COCC12 38521,C1(C(=O)NC(c2cc(F)ccc2OC)CC)CC2(CCC(N)CC2)C1 38522,c1(OC)cc(C(N2CCC(O)(CN(C(=O)CCc3ccoc3)C)C2)=O)cc(F)n1 38523,S(=O)(=O)(c1ccc(N2CCC3CCCC3C2)cc1Cl)NCC1N(C)CC(O)C1 38524,c1(OC)ccc(C)cc1CNC(=O)Nc1cccc(N2CCCCC2=O)c1 38525,Cc1nnccc1C(=O)NCCn1cc(C(=O)NC(C)CC2CCOC2)cn1 38526,C12(CNC(C(C)NC(=O)NC)=O)CC1CN(C(=O)C=Cc1c[nH]nc1C)C2 38527,c1(C(N(C(C)CNC(c2c(Cl)cnn2C)=O)CC)=O)cncc(F)c1Cl 38528,N1(C(C(C)c2cccs2)=O)CCC(N(CCCC)C=O)CC1.C1(C=O)C(C)C1(F)F 38529,CC1(C2CCN(C(=O)C(CN=[N+]=[N-])NC(c3cnco3)=O)CC2)CC1 38530,C1(C(N(CC(CC)OC)C)=O)C=CCN(C(C2(C)CC3CC3C2)=O)C1 38531,N1(C(C(=O)N2CC(C(CC)CC)C2)CCO)CCc2sccc2C1 38532,N1(CCCC(=O)NCC2N(C(C(CC)CC)=O)CCOC2)C(=O)CN(C)C1=O 38533,C1(C(N(CCC(C)NC(c2cc(-c3ccns3)on2)=O)C)=O)CC(O)CN1C 38534,Cc1c(C(N2CCC(CCNC(c3cc(O)cs3)=O)C2)=O)cnc2ccccc12 38535,S(=O)(=O)(C1CC2C(C1)C2(F)F)N1CCC(N(C2CCCC2)C)C1 38536,c1(C(=O)NC(CNC(CC(CCC)C)=O)C(C)(C)C)ccc(C)c([N+](=O)[O-])c1 38537,C(CCCCNC(=O)C(C)NC(=O)C1CC1)NC(C(C1CCOCC1)OCC)=O 38538,C1(NC(c2cc([N+](=O)[O-])n[nH]2)=O)CCN(C(=O)COCC2CC2)CC1F 38539,N1(C(c2ccc(C(C)=O)o2)=O)CCC(O)(CCNC(C2CCNC2=O)=O)CC1 38540,C1(NC(C(C)SCC)=O)CCCN(C(C23CC(CC)(C2)C3)=O)C1 38541,N1(C(C=C2CCC(C)CC2)=O)CCC2CN(C(c3cccc4nonc34)=O)C2C1 38542,CC1CN(C(=O)C(CO)NC(=O)Cc2ncccc2F)CC1(F)F 38543,c1(C(N(C)C)=O)cn(CC(N2CCC(CN(C)C(C3(C)CCCC3)=O)C2)=O)nn1 38544,N1(C(C2(C)C(C(=O)OC)C2)=O)CCOC(CCNC(=O)CCNS(C)(=O)=O)C1 38545,c1(C(=O)NCC(CN(C(COCCOCC)=O)C)O)c(N)ccc(C)c1F 38546,C1(=CCNC(c2cc(CCC)on2)=O)CCN(C(=O)C(C)(COC)OC)CC1 38547,C=CC1CCCCN1C(=O)COC(C1CCN(C(=O)OCC(C)(C)C)CC1)=O 38548,N1(C(CCC2CCN(C(C3N(CCC)CCC3)=O)C2)=O)CCC(O)CC(C)C1 38549,C(C(C)(C)C(=O)NOCc1ccc(F)cc1)NC(CCC1CCC(C)O1)=O 38550,N1(C(C(=O)N(CC(C)C)CCOC)=O)CCCC(C(C)C)CC1 38551,N1(C(c2c(CC)c(F)ccc2)=O)CCC2(CCN(C(C3CCC(C)O3)=O)CC2)C1 38552,N1(C(COCC(=O)OC)=O)CCN(C(=O)CC2(C(F)(F)F)CCC2)CCC1C 38553,CCC(CC(=O)NC(C(N1CC(C2=NOCC2)C1)=O)c1ccoc1)CC(C)C 38554,N1(C(C(CC2CC2)OC)=O)CCN(C(=O)Cc2cnn(C)c2C)CC(C)C1 38555,c1(C(=O)NC2CC(C)N(C(c3cncc(F)c3Cl)=O)C2)cccc2c[nH]nc12 38556,Cc1csc2c(C(=O)NC3(C4CCCN(C(C5(Br)CC5)=O)C4)CC3)ncnc12 38557,N1(C(CCSCC)=O)C2CCC1CC(O)(CNC(=O)C(F)Cc1ccccc1)C2 38558,C1(CNC(CCc2c(C)ncs2)=O)CCC2CN(C(=O)CC3(C)CC3)CCC2C1 38559,C(C(=O)NC1(C(=O)OC)CC1)(C(C)C)OCC.C12CCCCC1C(=O)NC2 38560,Cc1cc(C(C)(C)C)ccc1C(=O)NC1C=CCN(C(=O)C#CC2CC2)C1 38561,c1(CC(=O)NC2C3CCN(C(c4nc(C)oc4)=O)C32)c(C)cccc1C 38562,C1(COC)(NC(=O)CCC2CCCCC2)CCN(C(=O)C#CC(C)(C)C)CC1 38563,C1(CCC)(CNC(C2CN3CCC2C3)=O)CCN(C(c2[nH]ccc2COC)=O)C1 38564,c1(C(=O)NCC2N(C(C34CC(C)C3C4)=O)CC2)cccc(Cn2cncn2)c1 38565,c1(C(=O)NC(CCNC(C2CCC(C(=O)OC)C2)=O)(C)C)nc(C)sc1Br 38566,S(=O)(=O)(c1ccsc1C(=O)O)NCc1ccc(N2CCCC(C)C2)nc1 38567,C1(C(N(C(C)CC(=O)NCC(O)(C2CC2)C2CC2)C)=O)CC12CCOC2 38568,CC(CCCCNC(C1(NC(C23COCC2C3)=O)CCOCC1)=O)N(C)C 38569,C1(NC(c2nnnn2CCSC)(CC)C2CCOC2)CCC2(CC1)CSC2 38570,c1(C(=O)NC2C(NC(C(N(C)C)C3CC3)=O)CC2)ccc2cccc(Cl)c2n1 38571,c1(N(CCCOC)C(c2coc(-c3ccccn3)n2)=O)nccc(C)n1 38572,Cc1nc(C=CC(N2CC(NC(=O)CC3CCCCCO3)C(F)C2)=O)[nH]c1C 38573,C(=O)(CCC)N(CCCN(C(C)C)C(c1cnc(Cl)[nH]1)=O)CCO.C(=O)C1CC1 38574,CC(C(=O)N1CCOCC(CNC(=O)CNC(C2CCOCC2)=O)C1)S(C)(=O)=O 38575,C1(C(N2CC(CCNC(C3(C)CC3(C)C)=O)(OC)C2)=O)CN2CCN1C(C)C2 38576,c1(N2CC(C)(C)N(CCO)CC2)nc(N2CC3(C)CCC3(C)C2)c2ncsc2n1 38577,CC1CCN(C(c2ccc(O)nc2)=O)CC1NC(c1cnc(C(C)(F)F)s1)=O 38578,c1(C(=O)NC2(C3CCCCN3C(=O)C(F)=C3CCC3)CC2)cc(Cl)c(F)c(Cl)c1 38579,c1(C(N2CCC(N(C(c3ncc(CC)nc3)=O)C)CC2)=O)c(C)oc(C)c1C 38580,C1(NC(C2CCCC(C)C2)=O)C2CC3C1C3C2C(=O)NCCCC(F)(F)F 38581,c1(N2CC(C)(CNC(CCC(=O)N(CC)CC)=O)OCC2)ncnc2scnc12 38582,N1(C(C2CC(=C)C2)=O)CC2CC1CN(C(=O)CC1CC3CCC1C3)C2 38583,c1(CC)ncc(C(=O)NC2CC(N(C)C(c3c[nH]c(C(=O)OC)c3)=O)C2)[nH]1 38584,C1(CN(C(=O)CC2CCCO2)C)COCCN1C(C1(C)COC1)=O 38585,Cc1cc(=NCC2(O)CC3CCC2C3)[nH]c(N(C)CCOc2cccc(Cl)c2)n1 38586,CCC(CC(=O)N(CCNC(c1c(C)nnn1CC)=O)C1CC1)C(C)(C)C 38587,C1(CCCCNC(=O)CC2COCCO2)CCN(C(=O)CC2C=CCC2)CC1 38588,c1(C)c(C(C)C)cnn1C.C12CCN(C1)N2C(C(C)OCCOC)=O 38589,N1(C(c2cc(C)c(C)nc2C)=O)CC(CO)C2(CCN(C(=O)CC(C)F)CC2)C1 38590,C1(NC(c2c(C)onc2CO)=O)CC2CC1N(C(=O)C(=CC1CCCCC1)F)C2 38591,C1(c2n(CCC)nnn2)(N)CSC(C)C1.c1(CCCOC2CCCC2)ccccc1C 38592,c1(C(=O)NCC(c2c(C)nco2)=O)cccc(C(N)=O)c1 38593,N1(C(N2CCc3cccnc3C2)=O)Cc2cc(Br)ccc2C2CC1C2 38594,c1(CCC(=O)N(CCC)CCNC(C2CC3CC2C3)=O)ccc2c(c1)CCCO2 38595,c1(C(=O)OC(C(=O)N(C(C)C2CC2)C)C)nc(C(F)(F)F)cs1 38596,CC1(C)Cc2cccc(NCCCNC(=NCCCCl)NC3CC3COC)c2O1 38597,N1(C(C(CC)(C)O)=O)CC2(CC2)CC1C(=O)Nc1ncc(Br)nc1C 38598,C#CCC(C(=O)NCc1cncn1C(C)C)NC(=O)CNC(N)=O 38599,N1(C(c2cnc(C(C)C)[nH]2)=O)CC2C(N(C(=O)COc3ccc(Cl)cn3)C)C2C1 38600,C=CC(C)(CCOC)C(=O)NC1CN(C(c2sc(C)cc2Cl)=O)CC1SC 38601,C1(NC(COCCNC(COCCC=C)=O)=O)CCC(C(C)O)CC1 38602,C1(CN(C(Cc2ccn(CC)n2)=O)C)CN(C(=O)C(c2nc(C)cs2)C)CCO1 38603,Cc1cccc(C(CNC(c2ncncc2C)=O)NC(c2cn[nH]c2)=O)c1 38604,C1(C(=O)Nc2c(CC)csc2)CCN(C(c2ccc(=O)n(C)c2)=O)C(C)(C)C1 38605,C(C(C)(CC(C)C)NC(=O)Cn1ccc([N+](=O)[O-])n1)NC(C1C(OC)CC1)=O 38606,CCC(C)CCCC(=O)NCCCC(C)(C)C(=O)N1CCC12CCCCC2 38607,c1(N2CCC(C)C2CNC(c2ccc[n+]([O-])c2)=O)nc(Cl)ncc1C(F)(F)F 38608,N1(C(c2c(C)ccs2)=O)CCCCC1C(=O)Nc1cccnc1C(N)=O 38609,c1(C(N2CC(NC(CC3(C)CC3)=O)C2)=O)ccc(-n2cnnc2)cc1 38610,N1(C(CCC2CCCC(=O)N2)=O)CCCN(C(C23CSC(C2)C3)=O)CC1 38611,c1(C(=O)NCCN(CCCN(C)C)C(=O)CC2CC=CCC2)csc(O)n1 38612,C1(CCC(=O)NC(CC#C)CC)CCCCN1C(=O)CCc1nccn1C 38613,Cc1csc2ncc(C(=O)NC34CCCC3N(C(=O)COCCC(C)C)CC4)n12 38614,C1(C(=O)NC2CC(NC(c3cc(Cl)cc(Cl)c3)=O)C2)CCN2CCCC2C1 38615,n1(CC)ccc(CC(=O)NC(Cn2ccnn2)C(=O)N2CCC2(C)CCO)n1 38616,Cc1ccc(C)c(N(C(c2nocc2C)C(=O)NC2CCOC2)CC(C)C)c1 38617,c1(C(N2CC(O)(C(C)NC(C(C)C3CC3)=O)C2)=O)c(O)cccc1O 38618,C1(OC)CCC(COC(=O)CN2CCCC(CN3CCOCC3=O)C2)CC1 38619,C1(C)(C(=O)NCCCCN(C)C(C2CC2c2ccccc2)=O)CC(C2CC2)=NO1 38620,CC1CCN(C(=O)Cc2cnns2)CC1NC(=O)C(=CC1CCCCC1)F 38621,c1(C(=O)NCc2c(C(N3C(C(C)C)CC3)=O)occ2)ccc2nccn2c1 38622,Cc1c(Cl)cc(NC(=O)C(N2CCCC(C(N3CCCC3)=O)C2)=O)cc1I 38623,C(CC(C)(C)C)(C(=O)N1CCC(CF)(NC(=O)CSC(F)(F)F)C1)OC 38624,C1(CNC(CC=CC)=O)COCCN(C(C2(C)CC=C(C)CC2)=O)C1 38625,C1(C(N2CC(NC(c3cnc(-c4cccs4)s3)=O)C2)=O)CCc2nncn2CC1 38626,Cc1ccc(CC(N2CCC(C(C)NC(=O)C(C)CCO)C2)=O)cc1 38627,c1(OC)nc(Cl)c(C(N2CC(CNC(=O)COC3CC3)CC2C)=O)s1 38628,c1(NC)cccc(OC)c1C(N1CC(CO)(NC(C2CC(O)C2)=O)C1)=O 38629,C1(CN(C(=O)CCCc2ccncc2)CC)CCCN1C(=O)CCCC1CC1 38630,Cc1nn(C(C)C)c(C)c1C(N1CC2CN(Cc3ccc(C#N)cc3)C2C1)=O 38631,C12(C(N3CCN(C(C(C)=C(C)C)=O)C(CC(F)F)C3)=O)CCC(N=[N+]=[N-])C1C2 38632,N1(C(Cc2cc(C)no2)=O)CC(CNC(=O)CCCc2cnn[nH]2)C(C(F)(F)F)C1 38633,c1(CC)cccnc1C(=O)NC1CCC1CNC(c1ccn(CC(F)(F)F)n1)=O 38634,Fc1cc(SCNC(=O)CCC2CC(Cc3ccccc3)CN2)ccc1Br 38635,CCCCC(O)C(=O)NCC(C(C)C)NC(c1cnn(CCOCC)c1)=O 38636,c1(OC)ccc(NC(C2CC2C2CN(C(=O)Cn3nccc3C)C2)=O)cc1C 38637,c1(OC)cc(C(=O)NCC2(NC(C3CCN(C)C3C)=O)CCOC2)ncn1 38638,C1(C)(NC(c2c(COC)cccn2)=O)CCCN(C(=O)C(c2cccnc2)O)C1 38639,C(C(C)(O)CC(=O)NCCNC(=O)CNC(c1ccoc1C)=O)OC 38640,C(=O)(C(CCC)C(=O)NCC)NC(CCCC)C(=O)O 38641,CCCC(C#N)C(=O)NCCN(C(=O)C(CSC)OC)C(C)C 38642,N1(C(c2c(C)c(N)cnc2)=O)CC2CCCC2(NC(=O)Cc2ccccc2Cl)C1 38643,N1(C(=O)OC(C)(C)C)CCC(N2CCSCC2NC(=O)OC(C)(C)C)CC12CC2 38644,C1(NC(CCC=CC(C)C)=O)CC(C(=O)NCCN2CCCNC2=O)C1(C)C 38645,c1(OC)ncnc(C)c1C(N1CC(C(C)NC(=O)CCCCC2CC2)C1)=O 38646,c1(NC(C2(O)CCN(Cc3c(C)cccc3Cl)C2)=O)cc(F)cnc1C#N 38647,C=CCCCCCCC(=O)NCC(C)NC(c1c(N)cc(F)cc1F)=O 38648,c1(C(=O)NCC(CO)NC(C(C2CC(F)(F)C2)OC)=O)ccc(C(C)C)cc1N 38649,c1(NC(=O)C(C2CCCO2)C2CC2)cc(Cl)cc([N+](=O)[O-])c1O 38650,CC1CC2(CCN(C(=O)CC3CCCCO3)CC2)CN1C(c1nn[nH]c1Cl)=O 38651,c1(C(N2CC=CC(NC(c3cc(OC)ncn3)=O)C2)=O)cc2cccc(Cl)c2o1 38652,c1(C(N(CCC)CCNC(C2CCC2C)=O)=O)coc2ccc(OC)cc12 38653,C(C(=O)NN1CCSCC1)(C1CCS(=O)(=O)C1)NC(=O)OC(C)(C)C 38654,c1(CC)c(OC)cccc1C(=O)NC(CNC(C1COCCC1(F)F)=O)C(C)C 38655,N1(CCN(C(=O)CC2(N3CCCC3)CC2)CCNC(=O)C2CC2)CC2CC2C1 38656,N1(C(c2n[nH]c(O)n2)=O)CCC2(CCCN(C(c3ccc(Cl)nc3O)=O)C2)CC1 38657,N1(C(C(C2CCOC2)OCC)=O)CC2(CCCC2NC(=O)CC2CC2)C1 38658,N1(C(CC(C(F)F)OC)=O)CC2COCC2(COC)C1 38659,c1(OC)cc(OC)c(C(N2CCN(Cc3cccnc3Br)C3CC23)=O)cc1Br 38660,CCC(CC(F)F)C(=O)NC1CCCCN(C(C2CCCN(CC(C)C)C2)=O)C1 38661,CCCCC(C(=O)NCC1CC(OCC)C1)NC(c1ccoc1CC)=O 38662,Cc1ccc(Cl)c(O)c1C(=O)NCCCCC(C)NC(c1c[nH]nc1C)=O 38663,N1(C(=O)C2=CCCC2)CCC2C(CCCN2C(c2cnc(-c3ccco3)s2)=O)C1 38664,c1(C(=O)NCC(C)CN(C)C(C2CC(C(C)(C)C)=NO2)=O)ccc2n[nH]cc2n1 38665,C(c1cnc(C)nc1O)=CC(N1CC(C)CC(NC(CCCCC=C)=O)C1)=O 38666,c1(C(=O)NC2CCN(Cc3c(C)ccs3)CC2)cc(F)cc(Cl)c1 38667,c1(CC(N2CCC(C(=O)NC(C(=O)OC)C3CCC3)C2)=O)ccnc(O)c1 38668,C12(OC)CCCCC(C(=O)N(CC(C)NC(=O)CCn3ccccc3=O)C)(C1)C2 38669,C1(C)(NC(CCSC)=O)CCN(C(=O)C(C(C)C)c2cnc(C)s2)CC1 38670,c1(NC(Cc2cccc(C(C)N)n2)=O)cc(Br)c(F)cc1F 38671,c1(C(N2CCC(CC3CCC3)C2)C(=O)Nc2nnn(C)n2)cccc(OCF)c1 38672,c1(C(N2C(C3CCN(C(C(CC=C)C)=O)C3)CCC2)=O)ccc(C)c2cccnc12 38673,N1(C(CC2C(C)(C)C2)=O)CCC(NC(c2cc(N)c(O)c(F)c2)=O)C(F)(F)CC1 38674,C1(F)(C(N(C2CCN(C(C(C)(F)F)=O)C2)Cc2ccccc2)=O)CCCOC1 38675,CN1CCC2CN(C(C3CCN(C(c4cc(Cl)ncn4)=O)CC3O)=O)CC2C1 38676,N1(C(CNC(C(CC)C)=O)=O)CC=C(C(=O)NCC(O)Cn2cccn2)C1 38677,Cc1nc(Cl)[nH]c(=NCC2CC(CNC(=O)CC3CCCCO3)CO2)c1Cl 38678,C1(NC(C(c2n(C)cnc2)O)=O)CC2(CCC(NC(C3(C)CC3(F)F)=O)CC2)C1 38679,c1(C(=O)NCCN(C(c2c(C)snn2)=O)CC2CC2)csc2cc(Cl)cnc12 38680,C=C(C)CC(C)C(=O)NC1CCN(C(=O)C(c2cccc(OC)n2)(F)F)CC1 38681,c1(CC)cc(C(N2CCC(NC(c3cc(O)ncn3)=O)C2)=O)ccn1 38682,Cc1cc([N+](=O)[O-])c(Cl)cc1S(=O)(=O)CNC1(C(=O)O)CC2(C1)OCCO2 38683,n1(CCC)cc(Cl)c(C(=O)NC23CC2CN(C(=O)C(C)CC)C3)n1 38684,c1(COC)nccc(=NC2CCC3CN(C(c4n[nH]c(C)c4O)=O)CC23)[nH]1 38685,Cc1nnc2n1CC(C(=O)NCC1CCC1NC(=O)C=CCO)C2 38686,C(=O)(CCCC(C)(C)NC(c1n[nH]c(C)c1O)=O)N1CCC(OC)C(C)C1 38687,C(=O)(C(C)(C)S(C)(=O)=O)NC(CC1CN(C(Cn2c(=O)ccc(C)n2)=O)C1)C 38688,N(C1CCCn2cnnc21)C(CC(C)N(C(C(C1CCCCC1)C)=O)C)=O 38689,c1(C(N(C(C)CNC(C2CC=CCO2)=O)CC)=O)cc(Cl)c(N)cc1F 38690,c1(OC)ccc(C(CCO)NCC2CCC3(CC3)C2)cc1 38691,N1(CC2CCN(C(c3cc(OC)cc(F)c3)C)CC2)CC2CCC(OC)C2C1 38692,C(=O)(C1COc2ccc(F)cc21)N(C1CCN(C)C1)CC(=O)OC 38693,N1(C(CCSCC)=O)CCC(CNC(c2cnnc(C3CC3)c2)=O)C(F)(F)CC1 38694,C1(C)(COC)CCCN(C(=O)Cn2cc(CNC(C3(C#N)CC3C)=O)nn2)C1 38695,C1(C(C)NC(CCCOC(C)=O)=O)CCCN(C(=O)C(N2CCCC(O)C2)C)C1 38696,C(=O)(CCCCC(C)(C)C)N1CCC(NC(c2c(CC(C)C)onc2)=O)C1 38697,c1(OCC)cc(C(=O)NC2CCC(O)CC2)c(-c2nccs2)cn1 38698,N1(C(COC2C(CC)CCCC2)=O)CCN(C(c2ccnnc2O)=O)CC1C 38699,C(CCCCCC(=O)NC1CC1)n1ncc(NC(=O)Cn2cccn2)c1 38700,C(=O)(C1=C(C)S(=O)(=O)CC1)N1CC(NC(CCCC)=O)C(OC)C1 38701,N1(C(C2C(=C)C2)=O)CCC2(CCCCN(C(C3CC4CCC(C3)C4(F)F)=O)C2)C1 38702,N1(C(C(C)=C(C)C)=O)CC(C(=O)NCC(C)C#N)OC(C)C1 38703,N1(C(CCN(C)CC)=O)CCC(C2CCCN(C(C3C4CCCC34)=O)CC2)CC1 38704,N1(C(c2c(C)[nH][nH]c2=N)=O)CC2(CC(NC(=O)Cc3cn[nH]c3)c3nccn32)C1 38705,C(=O)(C#CC(C)(C)C)N1CC(OC)C(NC(c2ccccc2SC(C)C)=O)C1 38706,c1(CC)nn(C)c(C(c2nnnn2C(C)C)NCCCC(C)(C)OC)c1Cl 38707,N#Cc1c[nH]c(C(=O)NCCC2CC(NC(C3(n4ccnn4)CC3)=O)C2)c1 38708,C(CCCCC(=O)N1CC(O)CC1(C)C(=O)N(C)Cc1ccncn1)OCC 38709,c1(C(N2CCN(CCCNC(C3C(=C)C3)=O)CC2)=O)nn(C)cc1[N+](=O)[O-] 38710,C1(C2CCCN(C(c3ccn4nccc4n3)=O)C2)(NC(CC(C)SC)=O)CC1 38711,C12(C(=O)OC)CCCC1N(C(c1c(OC)cc(OC)cc1Br)=O)CC2 38712,N1(C(C(CC)OCC)=O)CCCC(C2CN(C(c3cccc4[nH]ncc34)=O)C2)C1 38713,Cn1cc(C2CC2C(=O)NC2CCN(C(C3(O)CCOC3)=O)C2)cn1 38714,c1(C(C)C)conc1CC(N1CC(CC(C)NC(c2c[nH]nc2C2CC2)=O)C1)=O 38715,C1(NC(C2(CCN=[N+]=[N-])CC2)=O)C=CCN(C(=O)CSc2cn[nH]c2)C1 38716,N1(C(C2C(=C)C2)=O)CCC2(CCC2)C(NC(=O)CCOc2cccc(Cl)c2Cl)C1 38717,N1(C(CCCc2nnc(C)n2C)=O)CCCC(NC(=O)CC2CCCCC2)C1C 38718,c1(CC)ccc2c(c1)OCO2.c12cccc(c1)N(C(C)=O)C2 38719,c1(N(C)C)nc2cc(C(=O)NC3CC(C)(NC(C4CC45CCC5)=O)C3)ccc2o1 38720,CCCC(CCC)CC(=O)NC(CCC1CC1)C(=O)N1CCC1CC(=O)NC 38721,N1(C(c2cc(C)c(F)cc2)=O)CCC2CCN(C(C3CCCCNC3=O)=O)C2C1 38722,c1(C(C)=O)ccc(C(=O)N(C2(C)CC(NC(=O)CC3CCC3)C2)C2COC2)cc1 38723,N1(C(C(C(C)O)N(C)C)=O)CCOCC(C)(CNC(c2coc(CO)c2)=O)C1 38724,c1(C(CNC(c2ccc(OCCOC)nc2)=O)C)ccc2cc[nH]c2c1 38725,C(C)(CNC(C1(C(C)(C)C)CCCCC1)=O)(C(C)C)NC(Cc1nnc(C)o1)=O 38726,C(=O)(C(C)(C)CCCNC(=O)C(F)C1CCOC1)NC(C)Cn1cnnc1 38727,N1(C(C2CN(C(C(CC)(C)COC)=O)CC(C)C2)=O)CCOC2C(O)CC12 38728,CC(CO)CCCNC(C1CCCN(C(=O)Cc2cccc(O)c2)C1)=O 38729,C(=O)(CCCCC(C)C)N1CCC(OC)(CNC(C2CCCC2O)=O)CC1 38730,C1(C(N(C(CNC(C2N(CC#C)CCC2)=O)C)C)=O)CCc2nncn2C1 38731,C(=O)(C1=NN(C)C(=O)CC1)NC1CCN(C(CC)=O)C(C2CC2)C1 38732,c1(C(N2CCC(COCC)C2)=O)cncc(-c2cccc(CC#N)c2)n1 38733,C(Cn1cncn1)(C(=O)N(C)C(C1CCOCC1)C)NC(C1C(=C)C1)=O 38734,N1(C(=O)Nc2nccc(OCC)c2)CCCN(CC2CC2)CC1 38735,C1(C(=O)NC2CC(CNC(CCc3cc(C)n(C)n3)=O)C2)OC(C)(C)OC1(C)C 38736,N1(CC(=O)N(c2cc(C(F)F)ncn2)CCO)CCC(C(F)(F)F)CC1.C(F)(F)F 38737,C=CCC(CNC(=O)CCn1cc(C(=O)OC)cn1)NC(C1(CC)CCOC1)=O 38738,C1(C)(C(=O)NC2CCC(C)N(C(C3C=CCCC3)=O)C2)Cc2ccccc2C1 38739,C1(C)(CNC(C(C2CC=CCC2)NC(CN(CCOC)C)=O)=O)CCCO1 38740,Cc1ccc(C(N2CC=CC(NC(=O)CCC3CCN(C)CC3)C2)=O)c(Cl)c1C 38741,C1(NC(=O)NCCC=CCCCCC)C2CN(Cc3ccccc3)CC12 38742,c1(C(=O)NC(CNC(c2ccc(C)cn2)=O)(C)C)cc(C2CCC2)n(C)c1C 38743,Cc1nnc(N2CCCC2c2csc(C)n2)n1CC1CCN(C(C)(C)C)CC1 38744,C(=O)(CC1COc2ccccc21)NC1CCN(C(C(=O)NC(C)C)=O)CC1F 38745,O(NC(=O)CC1(C(=O)C(C=CC)=O)CCCC1)CCOC(c1ccns1)=O 38746,N1(C(c2n(CC)nnc2)=O)C2CCC(C(=O)NC3CCCCCC3F)C1CC2 38747,c1(OC)c[nH]c(C(=O)NC(C2CCN(C(C3CCC4(CC4)C3)=O)CC2)C)cc1=O 38748,c1(C(=O)Nc2cc(C(=O)NCCC3CC(O)C3)ncc2)ccc(F)cc1F 38749,C(CC(O)C(=O)NC1CCCC1NC(C1(C2CCCO2)CC1)=O)N(C)C 38750,c1(C(=O)NCCCCNC(CCC#CC)=O)cc2ccc(C(C)=O)cc2[nH]1 38751,N1(C(C(COC)O)=O)CCCC(CO)(NC(C2CCC(F)(F)CC2)=O)C1 38752,c1(OC)cccc(C(CF)NC(=O)Nc2cnc(C3(C)OCCO3)s2)c1 38753,C1(C(N2CCC(CN(C)C(c3ncc(F)cc3N)=O)CC2)=O)CCCC(F)(F)C1 38754,CC1(C)CN(C(=O)CCCCC2CCCC2)CC1NC(c1cnn(C(F)F)c1)=O 38755,C(=O)(N=c1[nH][nH]c(C)c1Cl)C1(F)CN(C(c2c(NC(C)=O)cc(F)c(F)c2)=O)C1 38756,c1(C(C)C)ccc(C(=O)NCC2CC(F)(CNC(C3(C)CC3(F)Cl)=O)C2)cc1 38757,C1(c2nnnn2CCCF)(Nc2cccc(SC)c2)CCCC(F)(F)CC1 38758,c1(-c2occ(CC(C=C(C)C(F)F)=O)n2)ccc(OCC)nc1 38759,N1(C(Cc2ccc(C#C)cc2)=O)CC2CCC1CC2NC(c1c[nH]nc1CC)=O 38760,C1(CNC(C2(C)CCCC2)=O)CCCCCN1C(=O)C(F)CC1CCCC1 38761,c1(C(=O)NCc2c(C(N3C(CN(C)C)CCC3)=O)occ2)ccnnc1O 38762,c1(NC2C(=O)OCC23CC3)ccc(C(=O)O)cc1.C1(COCC)CCOCC1 38763,CC1CCN(C(C2CCCCC2O)=O)CC1CNC(C1(c2cccs2)CC1)=O 38764,C1(NC(C(C)=CC)=O)CC2(CCCN(C(C3CC3CCC)=O)C2)C1 38765,C1(C(N2CC(C(CC)CC)C2)=O)(NC(c2ccn(CCF)n2)=O)CCSC1 38766,Cc1ccc2sc(C(=O)N(CC(C)NC(c3cncc([N+](=O)[O-])c3)=O)C)cc2c1 38767,C1(C(=O)NCCCOCCNC(=O)C=CC2CCCO2)CC(C2CCCC2)C1 38768,C1(C(N(CCCNC(c2ncoc2C2CC2)=O)C2CC2)=O)CCCC(O)C1 38769,C(=O)(CCS(C)(=O)=O)N(CC(C)CNC(=O)CC1CCCC(C)C1)C 38770,N1(C(C2(CC#C)CCCC2)=O)CCC2(NC(=O)CCCOCC=C)CC2C1 38771,N1(C(C=C(COC)C)=O)CCCOC(CNC(=O)CC2CC3CCC2C3)C1 38772,C1(C(N2C(C3CCN(C(C4CCCN4C4CC4)=O)C3)CCC2)=O)CC(=O)N(O)C1 38773,c1(C(N(c2ccc(SC)c(C)c2)CCO)=O)n[nH]c2cc(-c3nccs3)ccc12.CN 38774,CC1(C)NC(=O)C2(CCN(C(=O)NCc3cc(C4CCC4)no3)CC2)O1 38775,C(=O)(CCC(C)CN(C)C)N1CCC(N(C(C(CC=C)C)=O)CC(C)C)CC1 38776,N1(C(CC2ON=C(C)C2)=O)CCC(C)(C)CC1C(=O)NC1CCC(C2CC2)C1 38777,CC1(c2nc(C3CC34CC4)nn2-c2ccc(Cl)nc2)CCCC(F)(F)C1 38778,c1(SCC)ccc(OC)cc1.N1(C(=O)OC)CCN(C(C2(n3cccn3)CC2)=O)CC1 38779,n1(CC)cc(NC(=O)CC(C)(C)N(C)C(c2cncc(C#N)c2)=O)ccc1=O 38780,C(C(=O)N=c1ccn(CCF)[nH]1)=CC(C)NC(C1CC2(CC2)CN1C)=O 38781,Cn1ncc(C(=O)NCC2CC(NC(c3ccc(O)nc3Cl)=O)C2)c1S(N)(=O)=O 38782,c1(NCc2cn(CC(C(=O)OC)O)nn2)cccc(C(=O)O)c1 38783,Cc1c(Cl)ccc(C(N2CCC23CN(C(=O)Cn2nc(Cl)ccc2=O)C3)=O)c1Cl 38784,C(=O)(CCC(C)(C)[N+](=O)[O-])NCC(C)CNC(=O)CSCc1ccccn1 38785,O=C1Nc2ccc(C(N3CC4CN(C(=O)CC5(O)CCC5)C4C3)=O)cc2C1=O 38786,N1(C(C(CC)N(C)C)=O)CCN(C(=O)C(N)=O)C(c2cn[nH]c2)C1 38787,C1(C2CCN(C(=O)CN3CCCC3C)CC2)(NC(CC(CC=C)(C)C)=O)CCC1 38788,C(CCCCC(=O)N1CCC(C)(C)C1C(=O)NC(C)C(=O)NC(C)C)SC 38789,CCC(O)C(F)(F)C(=O)N1CCC(CC(C)NC(=O)CCCn2ccnc2)CC1 38790,N1(C(CSCC)=O)CC(C)N(C(=O)Cc2csc(C(=O)OC)n2)CC1C 38791,C1(NC(Cn2c(=N)[nH]nc2)=O)CCC2(CCOCC2)C1 38792,Cc1ncc2ccc(C(N3CCC(CNC(C4(C5CC5)CC4)=O)C3)=O)cn12 38793,C1(NCC)COCCN(C(=O)COCn2nnc(C(=O)Oc3ccsn3)c2N)C1 38794,CCCC(C(=O)N(C)C)NC(=O)OC(C)(C)C.c12cnccc1O2 38795,N1(C(=O)Cn2ncccc2=O)CC2CCN(C(=O)C(Cl)=CCl)C2C1 38796,C1(C(=O)NC(C#C)CC2CC(NC(=O)CCCOCCOC)C2)OCCC1(C)C 38797,n1(C(C)C(=O)O)cc(C(C(=O)N(C)CCN(C)CCO)Sc2ccccc2)nn1 38798,c1(C2(C(=O)NCCC(C)(C)N(C)C(C3COCCO3)=O)CCC2)c(F)cccc1F 38799,CCC(CCCC(=O)NCC(C)CN(C)C)NC(=O)Cn1ccc(C)n1 38800,c1(CNC(c2ccc(CNC(c3cc(CC)[nH]n3)=O)cc2)=O)nnc2n1CCC2 38801,C1(COC)(N)CN(C(=O)C(C)=C(C)C)C1.C1(=O)CC1=O.C(C=C(C)C)N 38802,c1(C(=O)NCC2C(CNC(Cn3c(C)nnn3)=O)C2)ccc(NC=O)cc1 38803,C(=O)(CCCS(C)(=O)=O)N(CCCNC(c1ccc(F)c(C(F)F)c1)=O)C(C)C 38804,Cc1[nH]c2ccccc2c1C(=O)NCCC(C)NC(=O)CSC1CCCCO1 38805,N1(C(Cn2nnc(C)n2)=O)CCC2(CCCCC2NC(C2CCC(=O)N2C)=O)C1 38806,O=C(NN1CCSCC1)C(=O)N1CCCCC1c1ncc[nH]1 38807,C1(NC(c2ccnc3[nH]nnc23)=O)CC2(CCN(C(=O)C=CCO)C2)C1 38808,C(=O)(CC(C)CC(C)(C)C)NC1CC(CN(C2CCCC2)C(=O)COC)C1 38809,N1(CC(N2CC(F)(CNC(COCc3onc(CC)n3)=O)C2)=O)CC2C=CC1C2 38810,Cc1ccc(F)cc1CC(=O)NCC1(C)CCCN(C(C23CCN(CC2)CC3)=O)C1 38811,c1(SC)ccc(C(N2CC(NC(c3ccc(CN(C)C)[nH]3)=O)CC2C)=O)cn1 38812,C1(CCOC)(NC(=O)CC2CC2(Cl)Cl)CCN(C(=O)Cn2nnc(=O)[nH]2)CC1 38813,c1(SCC)nc(C)c(CC(=O)NC(C)(C)CCCNC(C2(C)CC2(F)Cl)=O)s1 38814,c1(NC(C2CN(S(CCC(=O)OC)(=O)=O)CC(F)C2)=O)ccc2c(n1)NC(=O)CC2 38815,c1(C(C)C(=O)NCC2CC(NC(c3occc3Br)=O)C2)cccc(C#N)c1 38816,CCC(O)(CC(=O)NCc1ccc(N2CCCC2)cc1C)c1ccccc1 38817,C(CC(CNC(=O)COC1CC=CC1)NC(C1CCCN1C(C)C)=O)OC 38818,C(=O)(C(C)C(O)CC)NCc1cc(C(=O)NCCC(=O)NCC)n[nH]1 38819,C1(CNC(c2cc3cc[nH]c3cn2)=O)CC2CCC1N(C(=O)Cc1cnoc1)C2 38820,C1(NC(=O)NCC(C)Oc2ccc(OC)cc2COC)CCCC(P(C)(C)=O)C1 38821,C(=O)(C(F)(F)C(C)(C)O)N1CC2C(NC(c3c(C)n(C)nc3)=O)(CC2)C1 38822,C1(C(=O)NCCOC2CCN(C(C3C(OCC)C3)=O)C2)CCC(C)CC1 38823,C1(C#N)(C(=O)NC(CC)CNC(C2CC(=O)N2)=O)CC12CCCC2 38824,N1(C(C(CC(C)C)F)=O)CC2C3CCC(C2C1)N(C(=O)CC1OCCC1(C)C)C3 38825,CC1CCC(NC(=O)CCC2CC2)CN1C(c1cc(-c2ccccc2)[nH]n1)=O 38826,c1(C(C(N2CCC(F)(CNC(C3CC=CC3)=O)C2)=O)O)cc(F)c(F)cc1F 38827,c1(C(=O)NC2CN(C(C3C(C)OCCO3)=O)CC2F)cn(C)c(=O)cn1 38828,n1(C(C)C(=O)NC2CCCC2NC(c2cncc(O)c2)=O)cnc2ccccc12 38829,Cc1nc2cc(C(=O)NC(CNC(C3CCCC(=O)N3C)=O)C(C)C)cnc2[nH]1 38830,C1(C(NOCC(C)O)=O)CCC(C2CC2)N1C(C1CCCC(O)C1)=O 38831,CC1CC(C(=O)N(C)CCOCCNC(=O)C(C)(C)C2CCCCC2)C1(C)C 38832,Cc1ccc(C=CC(=O)NCC2(F)CC(NC(C3CCSC(C)C3)=O)C2)cc1C 38833,CCCC(C)CC(=O)N1CCC(C(C)CNC(C2(CF)CC2)=O)CC1 38834,c1(C2C(C(=O)NCC3(O)CN(C(C(c4ccsc4)=O)=O)C3)CC2)ccc(F)cc1 38835,C(=O)(CC(F)F)NCC1CC(NC(C=C(C)I)=O)C1 38836,N1(C(C(CC)C)=O)CC2(CC(NC(=O)COc3c(C)cccc3C)C2)C1 38837,c1(NC(CC(=O)NC)C)nc(N2CCN(C3CCSC3)CC2)cc(C)n1 38838,c1(NC(N(C)Cc2ccc(OC)nc2)=O)ccc(F)cc1CC1CNC(=O)CO1 38839,c1(C(N2CCCC(N(C(C(CSC)O)=O)CCO)C2)=O)cc(F)ccc1F 38840,C(=O)(C1=CCCCC1C)NCC1N(C)CCN(C(c2cc(C)on2)=O)C1 38841,C1(COC)CCN(C(c2nc[nH]n2)=O)C(C(=O)N(CC(C2CCC2)OC)C)C1 38842,C1(C(N2CC(C(=O)OC)C2)=O)COCCC1NC(=O)CSC(C)C 38843,C1(NC(c2n(CC=C)ccc2)=O)CCCCC1N(C(=O)Cn1nccc1C)C 38844,c1(-c2n(CN(CC(=C)C)CC)ccn2)ccc(Cl)cc1 38845,C(C(COC)CC(=O)NC1CN(C(=O)CC(C)(C)O)C1)OC.[nH]1nnc(C(C)(C)C)n1 38846,C(CC(F)F)(C(=O)N1CCC(OC2CC2)C1)N(C)C(C1CC2C(C1)C2(F)F)=O 38847,c1(C(=O)NCC(CC)NC(=O)C=C(C)c2ccccc2)cc(C)cc([N+](=O)[O-])c1 38848,Cc1cc(C(N2CCC(C)(CCNC(c3ccnn3CC#N)=O)C2)=O)cc(C)c1 38849,c1(OCCC(=O)NC(C(C)NC(c2ccncc2)=O)C)ccc(CC#N)cc1 38850,C1(CNC(CC(=C)I)=O)CN(C(=O)CC)CC(C)O1 38851,c1(CC)cc(NC(c2coc(CNC(=O)CCC3CC3)c2)=O)cc(O)c1 38852,c1(C(N2CCCC(NC(c3cncc(SCC)n3)=O)C2)=O)ccc(N)c(Cl)c1O 38853,c1(N2CC(C(C)NC(=O)CCC3CC3(Cl)Cl)OCC2)cc(-n2cncn2)ncn1 38854,c1(C(C)=O)ccc(C(F)(F)F)nc1NC(C)(C)CNC(C1CC(C)OC1C)=O 38855,c1(-c2cc(NCc3c(C)c4c(s3)cccc4)ncc2)ccc2c(c1)OC(C)(C)O2 38856,C12CN(C(C3(O)CCN(C(=O)OC(C)(C)C)C3)=O)CCN1C2=O.C(C)(C)(C)OC 38857,C(C(F)(C(=O)NCCc1cocn1)C(C)C)NC(C(CC#C)O)=O 38858,c1(CC)cc(C(=O)NC2CCN(C(=O)CC3CC(C)=NO3)C2C(C)(C)C)n(C)n1 38859,Cc1cccc(C(C2CCCCC2)C(=O)Nc2cnccc2C)c1 38860,C(C(=O)NCC1CCCC(CNC(c2ccc(C#N)cn2)=O)C1)(C(C)(C)C)SC 38861,C(=O)(C(C(C)C)NC(c1ccccc1)=O)NC(c1c(C)scn1)c1ccccc1 38862,c1(COC)conc1C(=O)NCC1CCC(NC(C2CCN(C3COC3)C2)=O)C1 38863,Cc1c(C(=O)NC2CC(C)N(C(=O)CSc3nnnn3C)C2)noc1C1CC1 38864,Cc1c(C(C)NC(c2cnn(C)c2)C(=O)N(C)C)cccc1Cl 38865,N1(C(C2(CC#C)CCCO2)=O)CCC(C)N(C(=O)CC2(CC)CCC2)CC1 38866,C1(N(CCCC)C(C2CC2(F)Cl)=O)CCN(C(c2ccsn2)=O)CC1 38867,N1(C(C(C)O)=O)CC(F)(C(=O)NCCCn2cncn2)C1 38868,C(=O)(C(CCC1CCC1)NC(c1cnsc1)=O)NC1(CC(C)(C)C)CC1 38869,C=C(Br)CCC(=O)NC1CCN(C(c2cnccn2)=O)C1C 38870,N1(c2cc(C(C)(C)C)ncn2)CCC2CCC(C1)N2C(C1CCCO1)=O 38871,Cc1cc(Nc2cccn3cnnc23)ccc1[N+](=O)[O-].C12C3CN(CC13)C2=O 38872,N1(S(=O)(=O)CC2CC(CO)C3CC23)CCC(O)(C2(C(=O)O)CCC2)CC1 38873,C(C(C(=O)N(CC(=O)NC(C)C)C)C(C)C)NC(C1(CC=C)CCC1)=O 38874,Cc1ccc(C(N2CCN(C(=O)CC3=NNC(=O)C3)C3CC23)=O)c(F)c1F 38875,S(=O)(=O)(CCC(=O)NCC1CCN(C(c2cc(C)c(Br)o2)=O)CC1)NC 38876,CC1CN(C(=O)CN2CCN(C(C3CC3c3ccco3)=O)CC2)CC(C)(C)O1 38877,Cc1cnc(C(N2CCC(OCCO)CC2)C(=O)NCCC2CC2)c(C)c1 38878,c1(C(=O)NCC(C)(C2CCC2)NC(COC(C)C)=O)cn(CCO)nn1 38879,c1(CC(N2CC(CC(C)NC(c3ccc(C(N)=O)s3)=O)C2)=O)ccccc1O 38880,c1(C(C)NC(c2nnnn2CCF)c2ccns2)ccc(OCC#N)cc1 38881,c1(CC)cnc2cc(C(=O)NC3(CCC(=O)OC)CCCC3)[nH]c2c1 38882,c1(OCCC(C)C)ccc(C(=O)NCC(C)(C)NC(C2CCCN2C=O)=O)cc1 38883,c1(C(=O)NC2CC(C)N(C(=O)CC3(O)CCCC3)CC2)noc2cc(F)ccc12 38884,n1(CCNC(C(C)OCCC=C)=O)cc(N)cn1 38885,N1(C(C(COC(C)C)NC(Cc2c(C)nsc2)=O)=O)CCC2(CC2)C1 38886,C(=O)(CC(C)F)NCCC1(C(=O)NCCCC=C)CCC1 38887,C1(NC(=O)Cc2cncnc2)CCCC12CCN(C(c1ccc(Cl)c(Cl)c1)=O)C2 38888,c1(COC2CC(C(=O)OC)C2)cccc2c1CCC2 38889,c1(C(=O)NC2(CCOC)CCN(C(=O)C(C)=C(C)C)CC2)scc2c1CCCC2 38890,C1(CN(C(=O)CC2(OC)CCC2)CC)OCCC1c1n[nH]c(C)n1 38891,c1(C(N2CCN(C(=O)CC(F)F)C3CC23)=O)cc2ncc(Br)cc2o1 38892,Cc1[nH]c(=N)[nH]c1C(=O)Nc1ccc(CC(=O)N(C)C)cc1 38893,N1(C(c2c(C)n(C)nn2)=O)C2CCC(C2)C1C(=O)NC1CC(C(F)(F)F)C1 38894,C(=O)(CCCCC(=O)OC)N1C(CCNC(C(CC)C(C)O)=O)CCCC1 38895,C1(CCO)(CC)CN(C(=O)C(CO)NC(=O)CC2CC=CCC2)C1 38896,C(=O)(CCC(CF)CF)NC(C(=O)NCC1N(C(C)=O)CCC1)CC(C)C 38897,N(C(=NCC1CCSC1)NC1CCC1)Cc1cncs1 38898,c1(C(=O)NCCCC(C)NC(C2CC3CCC2C3)=O)cc2sccc2s1 38899,N1(C(CC2(C(=C)F)CCC2)=O)CCC2(CCC2)C(NC(c2cn(C)c(=O)n2C)=O)C1 38900,N1(C(C(CC)C(C)C)=O)CC(NC(c2ccc(C#N)c(C)c2)=O)CC12CCCC2 38901,CCCS(=O)(=O)C(C)C(=O)NC(C)(C)CN(C(=O)C=Cc1ncco1)C 38902,c1(SCCC(=O)NC2(CNC(C(CC)C)=O)CCOC2)c[nH]c2ccccc12 38903,CC(c1ccco1)=CC(=O)N(C1CCC(NC(=O)CC=CC(C)(C)C)C1)C 38904,C=C(C)CC(C(=O)NCCn1ccccc1=O)NC(=O)CCC=CCC 38905,Cn1ncc(C(N2CC3C(CNC(C4CCNC4=O)=O)C3C2)=O)c1-n1cccc1 38906,c1(C(C(=O)NC(Cc2c(OC)cccc2)C(C)C)OC)ccc(C#N)cc1 38907,C1(CCOC)(NC(c2ccc(Br)o2)=O)CCN(C(c2cccc(C(C)C)c2)=O)C1 38908,c1(-c2cn(CC3N(C(C4CCC(C)O4)=O)CCC3)nn2)cc(=O)cc[nH]1 38909,Cc1ncc(Cl)cc1N(C(c1[nH]c(C)c(C(=O)NC2CCCCC2)c1C)=O)C(C)C 38910,c1(C(N2CCC(C(C)(C)O)C2)C(=O)NC)cccc(S(N)(=O)=O)c1 38911,C=CCCCCCC(=O)NC(C)(CC)CCNC(C1COCCN1CC)=O 38912,N1(C(CCOCCOCC)=O)CC2(CCN(C(=O)CC3CCCC(C)C3)C2)C1 38913,c1(OC)ccc(C(N2CCN(C(=O)Nc3ccc(F)cc3)CC2)C2CC2Cl)cc1 38914,N1(C(c2c(CC)n(C)nc2)=O)CCC(C2CCN(C(=O)C3=CCCOC3)C2)C1 38915,CS(=O)(=O)C1CCN(C(C2(N)C3CCCCC23)=O)CC1 38916,c1(CNC(c2c(OC)csc2)=O)ccc(CNC(c2ccncc2)=O)cc1 38917,CSC1=C(C(=O)NC2CCN(C(=O)Cn3ccnn3)C(C)C2)CCCC1 38918,CCS(=O)CC(=O)NCC1CN(C(=O)C=CC(C)(C)C)CC1C(F)(F)F 38919,c1(CC)nonc1C(=O)NC(C)(CNC(c1ccncc1)=O)CO 38920,CC1(C(=O)NC2CCCC2(C)C)C=CCN1C(c1cc(CCO)on1)=O 38921,N1(C(c2ccc(CNC(CC(C)CN(C)C)=O)o2)=O)CC(CO)C(C)(C)C1 38922,c1(OC)c(F)ccc(F)c1C(N1CC(c2ocnc2CNC(=O)CCF)C1)=O 38923,C=CC1(C(N2CCC(C)(CNC(=O)Cc3cncnc3)C2)=O)CCCCC1 38924,C(=O)(CC1CCOc2ccccc21)NCC1N(C(C2CC(OC)C2)=O)CC(F)C1 38925,c1(C(=O)NC(CC(C)NC(=O)C=CC=C(Cl)Cl)C)cc2n(n1)CC1(CC1)C2 38926,Cc1cc(Cl)cc2cc(C(=O)N(c3cnn(-c4ccccc4)n3)C)[nH]c12 38927,C1(NC(C(CC)OC)=O)CN(C(c2cc(Cl)c(C)cn2)=O)C(C)(C)C1 38928,C1(C(=O)NCc2cc(CC)no2)CC(NC(=O)C(=O)N(C)C)C1(C)C 38929,c1(CCSCCC(N)C2CCC2)c(F)cccc1Cl 38930,CC1CC(NC(C2CC3CCC2O3)=O)CN(C(c2cccc(CF)c2)=O)C1 38931,c1(OC)cccc(C(=O)NC2CC(CNC(C3(CCO)CC3)=O)C23CCC3)c1O 38932,C1(OC)CCCN(C(=O)C(CNC(=O)CCc2ncnn2C)OC)CC1 38933,CC1(C)C2CCC1(C(N1CCC(NC(=O)Cn3cccn3)C(CO)C1)=O)C2 38934,N1(C(C(C)(C)F)=O)CCC(NC(=O)Cc2cc[nH]n2)C(F)C1 38935,N1(C(c2c(CC)c[nH]c2)=O)CC2CC(NC(=O)Cc3ccc(C(C)=O)s3)C1C2 38936,c1(C(=O)OC)cc(=NCC(C)(C2CC2)NC(=O)C=C(C)C(C)C)[nH]c(Cl)n1 38937,c1(C(N2CCCC2CF)C(=O)NCCCSC)cccnc1C(C)C 38938,Cc1ccc(CC(N2CCCC2c2cnco2)=O)o1 38939,c1(CC)ncccc1NC(=O)C(F)CC1CN(C(=O)C(C)OCC2CC2)C1 38940,C(c1cnccn1)=CC(=O)NC1C=CCN(C(=O)C(c2ccc(F)cc2)(F)F)C1 38941,c1(OC)ccc(N)c(C(=O)NC2CC(CNC(=O)C(C)C3CCC3)C(O)C2)c1 38942,CCCC(CCC)=CC(=O)NCCOC1CN(C(c2c(C)cnn2C(C)C)=O)C1 38943,C(=O)(C#CC1CCCCC1)N1C(C)(C(=O)NC2CC(C(C)C)OC2)CCC1 38944,O=C1CCC2(CN(C(=O)Cc3cc(Cl)ccc3Cl)C2)N1 38945,N1(C(c2[nH]ccc(=N)n2)=O)CC2CC1CC2CNC(=O)CC1CCCC1 38946,CCC(C)CCC(=O)N1CCCOC(C2CN(C(=O)C(CN(C)C)N(C)C)C2)C1 38947,CC(CC(N)=O)NC(C1C(CNC(c2nccs2)=O)C1(C)C)=O 38948,CN1C(=O)CCCC1C(=O)NCC1(CO)CCN(C(C2(C(N)=O)CC2)=O)C1 38949,c1(CC(=O)N(CC(C)N(C(c2ccc(COC)[nH]2)=O)C)C)cncc(C#N)c1 38950,CCC(CC)C(=O)NCCC(O)CNC(C1CCCC(C(=O)N(C)C)C1)=O 38951,C12(NC(CCC#C)=O)COC(C1)C(NC(=O)C(C)SCC)C2 38952,N1(C(CC(=C)C)=O)CCN(C(C2CCCCN2S(=O)(=O)CC)=O)C(CC)C1 38953,N#Cc1csc(CNC(=O)C(O)C2CN(C(=O)Cc3cncs3)C2)n1 38954,C1(COC)(NC(c2ccc(O)nc2)=O)CCCN(C(=O)C(O)P(C)(C)=O)C1 38955,c1(OC)cc(CC(=O)NC2CN(C(=O)CSC(C)C)CC2C)ccc1C 38956,C1(CNC(C(C=C)(C)O)=O)CC2(CCN(C(=O)CCCN=[N+]=[N-])C2)CO1 38957,N1(C(c2c(SC)cn(C)n2)=O)CC(NC(C2CC(C)CCO2)=O)CC(O)C1 38958,C(=O)(C(F)(F)CCn1cccn1)NC1C(NC(c2c(N)nccc2)=O)CCC1 38959,c1(NC(C)=O)ccc(Br)c(C(=O)NCCCNC(C2CC(C)=NO2)=O)c1 38960,c1(CCC)ncc(NC(C2CN(C(=O)CC(OCC)OCC)CC2F)=O)cn1 38961,c1(C(c2nnnn2C(C)(C)CC)Nc2cn(CC#C)nc2)snc(OC)c1Br 38962,N1(C(CC2CC(OC)C2)=O)CCCC2(C1)C(NC(c1nnsc1C)=O)CCN2C 38963,C1(F)(CNC(C2CCN(CC(C)C)C2)=O)CCC(NC(=O)Cc2c[nH]nc2O)C1 38964,Cc1nn2c(c1CNC(=O)C(O)c1ccco1)CN(C(C1CCCSC1)=O)CC2 38965,c1(C(=O)OC)cc(C(=O)NCCN(C(C2CCCC2O)=O)C(C)C)cs1 38966,CCC(C(=O)NCC1(C)CCN(C(=O)COc2ccsn2)CC1)C(F)(F)F 38967,N1(C(C2CN(C(C(C=C)OC)=O)CC2F)=O)CCCOCC1C 38968,c1(N2CCC(CC)C2)cc(=NCc2nc(=N)n(C)[nH]2)[nH]c(C(C)C)n1 38969,C1(C(N2CCCC(C)(CNC(C=C(C)C)=O)C2)=O)CC(c2cccnc2)=NO1 38970,N1(C(CSc2nc(C)[nH]n2)=O)CC2CN(C(c3nccn3C)=O)CC2C1 38971,Cc1cc(C(N2CCC(NC(C3(CO)CC3(F)F)=O)C2)=O)ccc1-n1ccnc1 38972,N1(C(c2c(Cl)cnc(CC)n2)=O)CCC(C2CCN(C(C3CC3CC)=O)CC2)C1 38973,N1(C(=O)NC(COC)C(C)C)CC2CS(=N)(=O)CC2C1 38974,C1(OC(C)C(=O)NCC(C)(C)NC(=O)CC2CC3(CC3)C2)CCCCC1 38975,C1(C(=O)NCCC2CC(NC(C=CCOC)=O)C2)Cc2nccn2C1 38976,c1(C(=O)NC(C(C)NC(=O)CC2(CO)CC2)C)ccc(Br)c(F)c1F 38977,CCC(C)CC(C)c1nc(-c2nc[nH]n2)nn1-c1cccnc1C 38978,N1(C(C2(C)C(C)C2)=O)CC2CCN(C(=O)CCc3ccc(C(C)(C)C)cc3)C2C1 38979,C1(NC(c2c(C)ccnc2C)=O)CC2CCC1C(NC(C1CCC(=O)N1C)=O)C2 38980,c1(C(=O)NC2CCC(NC(c3ccc(Cl)cc3F)=O)C2)c(Cl)ccc2c1OCO2 38981,C1(O)(CNC(c2ccc(CNC(c3cnc(=N)[nH]c3)=O)cc2)=O)CCCCCC1 38982,C1(NC(c2c(NC)scn2)=O)CN(C(=O)C(CO)OC)C(C)(C)C1 38983,c1(CC(N2CCC(O)(n3cc(CC4CC4)nn3)C2)=O)c(F)ccnc1F 38984,C1(C(=O)OC2CN(C(CCc3ccc(OC)nc3)=O)C2)CCC(C)NC1=O 38985,CC1=CC(C(C)(C)N(C2COCC2Oc2ccccc2)C2CC2)=C(C)S1=O 38986,C1(C(=O)NC(CC=CC)C(=O)NCC2(CCO)CC2)CCC2CC1CO2 38987,C(=O)(N=c1ccn(-c2cc(C)c(F)cc2Cl)[nH]1)c1c(OC)csc1 38988,Cc1cc(C(N2CCN(C(C34CSC(C3)C4)=O)CC2)=O)c(N)c(F)c1 38989,C1(C(N2CCC(NC(c3c(C(C)C)nns3)=O)CC2C)=O)CCCCC12CCC2 38990,n1(CC(N2CCN(C(c3c(C)cno3)=O)CC2CCO)=O)ncc2ncccc12 38991,Cc1ncc2n1CCN(C(=O)NCCCCOc1ccc(Cl)cc1)C2 38992,C1(O)(CNC(CC(=C)C)=O)CCCN(C(C2CCC3CC3CC2)=O)C1 38993,N1(C(c2cc(C)c(C)nc2O)=O)CC2CCN(C(c3ncsc3C)=O)CC(C2)C1 38994,O=S(=O)(c1ccc(Br)cc1Cl)NC(c1ccc(F)cc1)CN1CCC1 38995,c1(C(N2CC(C)(NC(C(n3ccc(C)n3)C)=O)C2)=O)ccc(C(C)=O)c(C)c1 38996,N1(C(C=C(C)Cl)=O)CCC2(CC1)CN(C(=O)Cc1cnn(C)c1)CC2CO 38997,c1(C(=O)NC2C(NC(CC3CC(=C)C3)=O)CCC2)cnncc1C 38998,C1(NC(c2nn[nH]c2Cl)=O)CC2(CCN(C(=O)Cn3cccc3)C2)C1 38999,C(=O)(C1=CC2(CCOC2)C1)N(C1CCN(C(c2ccoc2Br)=O)C1)C 39000,CCCC(C)(O)C(=O)NCCC1CN(C(=O)C(C)(C)C(=O)N(C)C)CCCO1 39001,N1(C(CC2ON=C(C)C2)=O)CCCCC1C(N1CCN(C(=O)C(C)C)CC1)=O 39002,C1(C)(C(N(CCNC(c2ccc(C(=O)CCC(C)C)s2)=O)CC)=O)CC(C)=NO1 39003,c1(C(N(CCCNC(C2(C)CCC(F)(F)C2)=O)C(C)C)=O)cnc2n1CCOC2 39004,c1(OCC(=O)NC2CCCCC2CNC(c2cnc(O)s2)=O)nc(O)nc(O)n1 39005,C#CCCC(O)C(=O)NCC1CCCN1C(c1ccccc1C(=O)OC)=O 39006,N1(C(CCC(=C)C)=O)CCCC(O)(CCNC(=O)C(O)C(C)CC)C1 39007,C(C)(C(C)NC(c1ncoc1CNC(=O)C=Cc1cncs1)=O)(C1CC1)OC 39008,c1(C(=O)NC(C(=O)NCC(C#C)OC)CCC)nn(C)cc1C#C 39009,C1(CNC(=O)C(F)C2CC2)CC2(CO1)CN(C(c1ccc3c(c1)CCC3)=O)C2 39010,C1(C(=O)NCC2(CC)CCOC2)CN(C(=O)CN2CCNC2=O)C(C)(C)C1 39011,CCC(C#N)C(=O)NCC1CCCC(NC(C2(C(F)(F)F)CCOCC2)=O)C1 39012,Cc1ccc(C(=O)N(C(C)CCNC(=O)C(F)C(C)(C)O)C)c(N)c1Cl 39013,C1(C2CCN(C(=O)C(F)(F)C3(OC)CCCC3)C2)(NC(CC(CCC)C)=O)CC1 39014,C1(C)(CNC(=O)NC2N(C(=O)OC(C)C)CCC2)CCC(=O)NC1 39015,n1(CC)cc(C(=O)NC2CC(CNC(c3ccc(O)cc3)=O)C2)c(C)n1 39016,N1(C(C(C)C2CC2)=O)CCc2ccc(C(N3CC(C)(C#N)C3)=O)nc2C1 39017,c1(C(N2CC(O)(CN(C(=O)CO)C)C2)=O)ccc(-c2cscn2)nc1 39018,C1(C(N(C2CCCCN(C(=O)C=CSc3nc[nH]n3)C2)C)=O)CC2C(C1)C2(C)C 39019,N1(c2ccnc(C)n2)CC2CC(NC(c3c(C)ncn3C)=O)C2C1 39020,N1(C(Cc2n[nH]c(=N)s2)=O)CCC(C2(NC(c3ccn4nnnc4c3)=O)CC2)C1 39021,c1(C(=O)NCC(C)(CC)NC(C(CC)OC)=O)cccc2oncc12 39022,O=C1CCCc2cc(C(N3CC(NC(c4cc(F)cc(F)c4Cl)=O)C3)=O)ccc21 39023,c1(C(N(C2C(C)CCNCC2)CC2CCOCC2)=O)ccc(S(C)(=O)=O)cc1 39024,c1(C(N2CCN(CCNC(CCC=C(C)C)=O)CC2)=O)ccc2nn[nH]c2c1O 39025,C1(C(N2CC(C(C)C)N(C(=O)CCC3CC3C)CC2)=O)CC2CCC(C1)N2C 39026,S(=O)(=O)(c1cccnc1NCc1ccc(C)s1)NC(CC)C(O)C(C)C 39027,CCCC(CC(=O)NCC1CCC(C)CC1)NC(c1sc(C)nc1C)=O 39028,C1(C)(CNC(c2c(C)cns2)=O)CCCN(C(c2ccc(C(C)C)cc2F)=O)C1 39029,c1(C(=O)NCC(C)(C2CCC2)NC(CS(=O)(=O)NC)=O)cccc(C#CCO)c1 39030,C=C(C)C(C)(C)C(=O)NCC(C1CCN(C(C2Cc3nnsc3S2)=O)CC1)C 39031,C1(CC)CCN(C(=O)COC2CCCOC2)C(NC(=O)CC(C)(C)CN(C)C)C1 39032,Cc1ccc(-n2ncc(C(=O)NC(c3cccnc3)C3CC3)n2)cc1 39033,N1(C(C(CC2CCC2)NC(C)=O)=O)CCCCC1C1C(C(=O)O)C1 39034,N1(C2CCN(C)C2=O)CCC2(CC1)CC2C(N1CCCC1c1ccc(O)cc1)=O 39035,c1(C(N2CC(O)(CNC(C(=O)NCCOC)=O)C2)=O)c(C)[nH]cc([N+](=O)[O-])c1=O 39036,C1(NC(C(c2cc(C)sc2)(F)F)=O)CN(C(=O)C2CC2)C2CCCCC12 39037,C(=O)(CC(C)F)N(C1CC(NC(C(C2CCCCC2)OC)=O)C1)C 39038,C1(NC(c2ccc(C#C)nc2)=O)C2CCCN(C(=O)C=CC(C)C)C2C1(C)C 39039,C1(CCNC(C(C2CCOC2)N(C(C2CCCC2)=O)CC)=O)CCC(C)(C)CC1 39040,C(=O)(n1ccc(C(=O)OCC2N(C(=O)C3CC3)CCCC2)n1)OC(C)(C)C 39041,C(=O)(CCCC(CC)CC)N1CCN(C(COCCCCOCC#C)=O)C(C)C1 39042,C(=O)(C1=CCN(C(=O)CC(C)(C)CN(C)C)CC1)N1CCCC(CC=CC)C1 39043,c1(C(N(CCC(C)(C)NC(C2CCCC(O)C2)=O)C)=O)nccc2[nH]ccc12 39044,C(C)(C(C(=O)NCc1ncc(F)cc1F)C(C)C)NC(C(F)=CCC)=O 39045,C(=O)(CC(C)(C)N(C)C)N(CCCCN(C(C(C)c1cc[nH]n1)=O)C)C 39046,N1(C(C2CC(C)(C(=O)OC)C2)=O)CC(NC(=O)C=CS(C)=O)C(F)C1 39047,CC1CCC(C(=O)NC2(CCNC(=O)Cc3cccnc3)CC2)O1 39048,c1(C(C)=O)ccc(C(=O)NCC(C)CN(c2ncnc(C)c2OC)C)c(F)c1 39049,N1(C(C2(CNC(c3cc4n(n3)CCO4)=O)CC2)=O)CC2COCC(C2)C1 39050,c1(C(N2CC(CC(C)(C)CC3CCO3)C2)=O)ccc(Cl)cn1.c12cccnc1C(O)CN2 39051,c1(C(=O)NCCCCc2cn(Cc3cnn[nH]3)nn2)onc2ccccc12 39052,N1(C(=O)Nc2cc(C)cc(C)c2)Cc2cccn2CC(C(N2CCSCC2)=O)C1 39053,c1(C(N(C2CCCC(N(C)C(=O)C3CC3)C2)C)=O)cc(-c2cccnc2)nn1C 39054,CCC(F)(F)CC(=O)N1CCC(F)CC1C(N1CCC(CN=[N+]=[N-])C1)=O 39055,C1(N(c2c(-n3cccn3)cc(OC)nn2)C2CC2)CCN2CCCCC12 39056,N12CCCOC(C1)C2=O.Cn1cc(OC2(CNC(=O)CCCN(C)C)CC2)cn1 39057,C(C)(C)(CCCCC(=O)NCC1CN(C(c2sccc2C#N)=O)C(C)(C)C1)OC 39058,CC(C)(CN1CCOCC1)C(=O)NC1CC(CCNC(C2(C3CC3)CC2)=O)C1 39059,C(C(C)(C)C(=O)NCC1CCC(C)(CC)O1)NC(C(C=C)C)=O 39060,CC(C)(CCF)C(=O)NC1C=CCN(C(c2cc(CCO)on2)=O)C1 39061,C1(CNC(C(C)=CC2CC2)=O)CCCC1C(=O)NCC(N1CC=CC1)=O 39062,N1(C(C23C(C)(C)OCC2C3)=O)CCCC2(C1)CN(C(c1ncc(F)cc1F)=O)C2 39063,c1(C(=O)NC2CC(C)(NC(C(CC)N(C)C)=O)C2)ccc(-c2cnco2)cc1 39064,c1(N2CCCC(CNC(C3(C)CC=CCC3)=O)C2)ccccc1C#N 39065,c1(C(N2C(COC)(CNC(=O)C(C)C(C)O)CCC2)=O)cc2[nH]nc(C)c2cn1 39066,c1(OC)ccc2[nH]c(=NCCS(C)=O)[nH]c(=NCCc3ccc(Br)cc3F)c2c1 39067,c1(C(N2CCC(NC(C3(Br)CCC3)=O)CC2)=O)ccc(Cl)c(F)c1F 39068,c1(C(=O)NC2C(C)C2C)cc(C#N)ccc1N 39069,Cc1ccc(CNC(=O)CN2CCC(CC(=O)N(C)Cc3ccccc3)C2)s1 39070,C#Cc1ccc(OCC(=O)NCCC2(NC(C3CCN(C)S3(=O)=O)=O)CC2)cc1 39071,c1(C(N2CC(NC(c3cccnc3)=O)C(C(F)F)C2)=O)cc(=O)n2nccc2[nH]1 39072,c1(C(=O)NC2C(CN(C(C(C)(C3CC3)NC(C)=O)=O)C)CCC2)nc(Cl)oc1C 39073,N1(C(CC(CC)OC)=O)CCOCC(C)(CNC(c2ccc(C)cc2SC)=O)C1 39074,CCCC(CCC)=CC(=O)NC(C)CC(C)NC(=O)CCc1nccn1C 39075,c1(CN(c2nnc(C(CC)(C)C)s2)C=O)ccc2nc(O)n(C3CCCC3)c2c1 39076,c1(CC)cc(C(=O)NC2CC(NC(C3(OCCNC(C)=O)CCCC3)=O)C2)no1 39077,C1(NC(c2n[nH]cc2I)=O)CC12CCN(Cc1c(O)cc(F)cc1F)CC2 39078,N#Cc1c(OCC(=O)NCC2CCCN2C(c2ccco2)=O)cccc1Br 39079,c1(CC)cc(C(=O)NC2C=CCN(C(C3CC(=O)N(CC)C3)=O)C2)c(C)nn1 39080,C(=O)(C(C(C)(C)C)OC)N(CC(=O)N(CC(N1CCCC1)C)C)CCOC 39081,C1(C)(CC(=O)N(CCCCC)C(C)C)CCN1C(=O)CN(CCCN=[N+]=[N-])C(C)C 39082,Cc1cnc(Cl)c(CNC2CC(C(=O)Nc3ccsc3C#N)C2)c1 39083,C1(OC)CCN(C(C2CCCCC2)C(=O)NCCCC2CC2)C1 39084,C(=O)(CS(C)(=O)=O)NC(C(C)NC(C1(C)CC(=C)C1)=O)CO 39085,N1(C(CCc2n(C)ccc2)=O)CCCN(C(C2CCCCO2)=O)CC1CO 39086,c1(C(c2ccc(Br)o2)NCC2C(CCC)C2)nnnn1C1COC1 39087,c1(C(N2CC(C)S(=O)(=O)CC2)=O)ccc(Nc2cccc(F)c2)c([N+](=O)[O-])c1 39088,C(=O)(CCC(=O)NC1C=CC(CNC(C2C(Cl)(Cl)C23CC3)=O)C1)NC 39089,C1(CN(C(=O)C2=CCC2)C)CCCCN1C(c1c[nH]c(-c2ccc(F)cc2)c1)=O 39090,c1(C(=O)NC2CC(C)(NC(=O)C3=COCCO3)C2)ccnc(S(N)(=O)=O)c1 39091,c1(C(=O)NC(CNC(c2nc(OCC)sn2)=O)(C)C)ccc(OC)c2ccsc12 39092,c1(CC(=O)NCC(C)CNC(=O)C(C)C(F)(F)F)cccc(C#N)c1 39093,C1(C(=O)OCCCOC)CCCCC1NCc1cccc(OCCC=C)c1 39094,N1(C(CCCC2C(C)C2)=O)CCC(C2CC2)C1C(=O)NOCCC(C)O 39095,c1(CNC(c2cccc(-n3c(C)c(C(=O)O)cn3)c2)=O)cn2cccc(C)c2n1 39096,N1(C(C(=O)NCc2n(CC)c(C)nc2)=O)CC2CCC2(C)C1 39097,C(=O)(C(=O)N=c1cc(C)o[nH]1)NCC(CC)NC(c1ccc2c(O)n[nH]c2c1)=O 39098,C(C)(N=c1nc2c(ncn2C)c(NC(C)CS(N)(=O)=O)[nH]1)c1n(CC)ncc1 39099,c1(C(N(c2nc(OC)c(F)cn2)C2CCCNC2)=O)cc(O)ccc1[N+](=O)[O-] 39100,c1(C(=O)NCCN(C(c2c(C)nc(CCCC)s2)=O)CC)cc2n(n1)CCOC2 39101,C(CCC(C(=O)NCCC(=O)OC(C)C)NC(=O)CCc1nc(C)no1)OC 39102,c1(C(=O)NC2C(CNC(=O)CCC3CC3)CCC2)ccc(C(F)(F)F)nc1O 39103,c1(C(=O)NCCC(=C)CNC(C2(c3ccccc3)CC2)=O)ccc(C)c(O)c1 39104,C(=O)(C(C)(C)CCCO)NCC1CC2CN(C(c3cccc(OC)n3)=O)CC21 39105,C1(C(=O)NCc2c(C)occ2)CN(C(=O)CCC(=O)C2CC2)CC12CC2 39106,C(=O)(C1=CC2CCC=CCCC12)NCC1C(C)CCN(C(C2(O)COC2)=O)C1 39107,CCC(CC)C(=O)N1CCCCC1C(=O)N(CCN1CCCC1=O)CC 39108,C(CC(C)(C)CC(=O)NCCCCC(C)NC(c1cc(C2CC2)n(C)n1)=O)OC 39109,Cc1ccnc(C)c1NC(C12CCC1CN(C(=O)Cc1c(C)nn(C)c1C)C2)=O 39110,C1(C(=O)OCC2CCCO2)(NCc2ccccc2C(F)(F)F)CCOCC1 39111,CC1CN(C(C2CCS(=O)(=O)N2)=O)CCN1Cc1cccnc1-c1ccccc1 39112,c1(CC(=O)NC(CNC(=O)C=CC2CCC2)C2CCC2)nc([N+](=O)[O-])n[nH]1 39113,C(=O)(CCCCCCC=C)N1CC(CC#C)(C(=O)NC2CC(=O)N(CCC)C2)C1 39114,N1(C(c2ccc(CNC(N)=O)s2)=O)CC2CC1CCC2O 39115,CC(C)CN=C(NCc1ccccc1CO)NC(C1CCOC1)C 39116,Cc1cnc(-c2cn(CCN(C(=O)CC(C)(C)C#N)C(C)C)nn2)c(C)c1 39117,Cc1scc(C(N2CC(NC(C3(C4CCCO4)CCCC3)=O)C(O)C2)=O)c1N 39118,c1(OCCC)ccc(CNC(=O)NC2CC(C(=O)OC)C2)cc1 39119,C1(CNC(C2CC(=C)C2)=O)CC(CNC(=O)Cc2cnn(CC(=O)NC)c2)CO1 39120,CC(C)C(C(=O)N1CC2CC1C2NC(=O)COCC1CC1)NC(=O)OC(C)(C)C 39121,C1(NC(C(CC=C)N(C)C)=O)CC2CC1CN(C(C1(COC)CCCCO1)=O)C2 39122,Cc1cnc(C#N)c(-c2c[nH]nc2C(=O)NCc2cc(F)c(F)cc2I)c1 39123,CC1C(NC(C2COCCN2C)=O)CCCN1C(c1[nH]ncc1C#N)=O 39124,N1(C(CC2(C#N)CC2)=O)CCN(C2CCCN(C(=O)Cc3c[nH]nc3O)C2)CC1 39125,CC1(C(=O)NCC2CN(C(=O)Cn3cc(C(F)(F)F)cn3)CC2O)CC=CCO1 39126,c1(CNC(=O)CC2CC=CCC2)ccc(C(N2CCC(c3cnn[nH]3)C2)=O)cc1 39127,C1(C)(COC(c2c(C)ccnc2C(C)C)=O)CC(C2CC2)=NO1 39128,c1(SC)ncccc1NC(=O)CCC1CCCN(C)C1 39129,C1(NC(=O)NC)CCN(C(=O)CCCN2CCOC2=O)C1 39130,c1(C(N2CCC(C)(CNC(C3CS(=O)(=O)C3)=O)C2)=O)c(F)ccc(Cl)c1N 39131,c1(C(N(CCCNC(C(C)SCC)=O)C2CC2)=O)cc(O)c2[nH]c(C)nc2c1 39132,C1(O)(CNC(CC2(CSC)CC2)=O)CCCN(C(c2c(Cl)nsc2Cl)=O)C1 39133,c1(C(C(N2CCC(C(F)F)(CNC(C)=O)C2)=O)C)ccccc1S(N)(=O)=O 39134,C1(NC(CCCC(=O)OC)=O)C2CC(CN(C(C3(CF)CC3(F)F)=O)C2)C1CO 39135,C1(NC(c2c(COC)scc2)=O)CCCCC1CNC(c1sc(C)cc1C)=O 39136,c1(CNC(c2cnc(SC)s2)=O)cc2n(n1)CCN(C(C1CC(C3CC3)C1)=O)C2 39137,N1(C(C2C=C(C)CS2)=O)C2CCC1CC(C(=O)NC(C)C(C)F)C2 39138,C1(CNC(C2ON=C(CC)C2)=O)CC2CCC1N2C(c1cc(C)ccc1C)=O 39139,N1(C(c2ncn(CC)c2)=O)CCC2(CCN(C(c3cnoc3CC(C)C)=O)C2)C1 39140,C1(OC(C)C(=O)NCC(C)(C)CNC(=O)COC2CC2)CCCCCC1 39141,c1(C(N2CCC(NC(c3c(C)onc3C(F)(F)F)=O)C2C)=O)ccc([N+](=O)[O-])[nH]1 39142,C1(C(=O)NC(C)CCCNC(c2c(C(F)(F)F)ncn2O)=O)CC(=O)OC1(C)C 39143,c1(C(CC)(C)C)cn(CC2CC(NC(=O)C(F)OC(F)(F)F)C2)nn1 39144,C1(C(N2CC(C)N(C(C3CS(=O)(=O)CCO3)=O)CC2)=O)Cc2nccnc2C1 39145,CC1=NNC(=O)C1CC(N1CCCCC1CNC(C1(c2ncco2)CC1)=O)=O 39146,CS(=O)(=O)C1CCN(C(C(=O)NCc2ccccc2)C2COC2)C1 39147,C(=O)(CC(CC(C)C)NC(=O)C(CCC)=CCC)NC1(CC=C)CC1 39148,CC1CCN(C(=O)C(=O)NCC2CCCN(C(C3CNC(=O)N3)=O)C2)CC1 39149,c1(C(=O)NC2C(C)CN(C(c3c[nH]nc3F)=O)C2)n[nH]c2c1CCCC2 39150,n1(C2CN(C(CC#C)=O)C2)ccc(=NC(=O)c2ccc(NC(N)=O)cc2)[nH]1 39151,c1(C(=O)OC)cccc(C(=O)NC(CO)C(C)NC(C2CCS(=O)(=O)N2)=O)c1 39152,C(=O)(CCS(=O)(=O)N(C)C)N(C(CNC(c1ccc(OCC)nc1)=O)C1CC1)C 39153,C1(C(=O)NCCCC(C)NC(c2sccc2CO)=O)CC2CC1CC2O 39154,C1(CNC(c2c(C)cc(C)[nH]2)=O)(NC(c2c(C)ccn2C)=O)CC2CCC1CC2 39155,Cn1cc2c(C(=O)NCCC3=CCN(C(=O)CSCC(N)=O)CC3)cccc2n1 39156,CC(C)CC(CC(C)C)NC(=O)CCCC(C)NC(=O)Cc1ccc[nH]1 39157,C12(CNC(c3ccc(C)nn3)=O)CC(NC(c3nc(Br)c[nH]3)=O)(C1)C(C)O2 39158,Cc1cc(C(=O)N(C)CCN(C(=O)C=Cc2ccco2)C)sc1C 39159,c1(C(=O)NC2CCN(C(CN(CCCCCC)C)=O)C2)cc(=O)c(OC)c[nH]1 39160,c1(C(=O)NC)ccnc(CN(C(c2cocn2)=O)CC2C3CNC2C3)c1 39161,c1(CSCC(C(C)(C)C)OC)nc2ccccc2o1 39162,C1(C(=O)NC2(CF)CN(C(CC3(C)CCC3)=O)C2)CNC(=O)CC1(C)C 39163,N1(CC(=O)NCC(CCOC)NC(=O)C(n2cc(Cl)cn2)C)CCCCCC1 39164,C12(C(=O)NC(CCCC)C)CCCC1CN(C(C1(COC)CC(=O)C1)=O)C2 39165,C1(C(C=CC(=O)OCC(COCC)O)=O)CCCN(C(C)=O)C1.C(=O)CC 39166,N1(C(C(Cn2ccnn2)NC(C2(CC)CC2)=O)=O)CCCN(C(C)=O)CC1 39167,Cc1cc(C(=O)NCC2CC2NC(=O)Cc2nc(C(C)C)c(C)s2)c(N)c(Cl)c1 39168,N1(C(CNC(=O)NC(c2nocc2N(C)C)C)C)CCN(C)CC1 39169,c1(C(N2C(CC=C)CCC2)=O)cn2c(n1)C(N)CCC2 39170,Cc1cccc(CN(C(c2ncccc2C)C(=O)NCCC2(C)CC2)C)c1Br 39171,Cc1nc(C)n(CCC(=O)NC(CO)C(C)NC(c2sc(N(C)C)nc2C)=O)n1 39172,c1(C(N(CCNC(C(C2CC2)OCC)=O)C)=O)nc(-c2ccccc2F)oc1C 39173,C1(C)(C(N2CCC(CCc3cn(C(CC)CC)nn3)CC2)=O)CCNC(=O)C1 39174,S(=O)(=O)(c1cccc(Br)c1)N1CCC(C#N)(NC(c2c(F)ccc(Cl)c2F)=O)C1 39175,CC1C(NC(=O)C=Cc2ccccc2)C(C)CCN1C(C1CCC=CO1)=O 39176,Cc1nc2ccc(-c3cncc(NS(C)(=O)=O)c3)cc2n1C 39177,N1(C(C2(COC)CC=CC2)=O)CC2CCC(C1)C2C(N1CCCC1CO)=O 39178,c1(C(N2CC(CCC)N(C(=O)CCN3CCCC3)CC2)=O)cc(O)cc(C#N)c1 39179,Cc1c(C(N2CC(CNC(C3(C)CCCC3)=O)C(C)(C)C2)=O)nn2ccccc12 39180,N1(C(CCOCC)=O)CC2C(CN(C)C(C3(CF)CC(F)(F)C3)=O)C2C1 39181,N1(C(c2nnc(O)nc2O)=O)CCC2CN(C(=O)C(O)CC(F)F)C2C1 39182,c1(C(=O)NCC2CN(C(CCCCSC)=O)CC2O)cc2cc(Cl)ccc2[nH]1 39183,C1(CNC(=O)C(=O)NC2CC2)CN(C(=O)CCC2OCCO2)CC12CCOCC2 39184,C(=O)(C(CC(F)F)c1ccccc1)NC1(C)CN(C(C2(C)N(C)CCC2)=O)C1 39185,O=C1NC(=O)C(CC(=O)NC23CC(C2)N(C(c2ccncc2O)=O)C3)N1 39186,N1(C(c2ccc(N)c(F)c2)=O)CC2ON=C(CNC(=O)CCc3nccs3)C2C1 39187,C1(C(C)C)C(=O)N1.N1(C2CN(NC(C)=O)C2)CCN(C(=O)CCC=C(C)C)CC1 39188,O=C1CN(CC(F)F)C(C(=O)NON2CCN(C(=O)CC3CCC3)CC2)CN1 39189,C1(C2CCN(C(=O)Cc3cnsc3)C2)(NC(C2C3COCC23)=O)CC1 39190,Cc1scc(C(=O)NC(Cn2cccn2)C(=O)NCC2([Si](C)(C)C)CC2)c1C 39191,c1(C(=O)NC2C(NC(C3CCCC(C)(C)C3)=O)COC2)nc2cc(O)ccc2[nH]1 39192,CC1CCCc2ncc(C(=O)NC3CN(C(C4CC5CC4C5)=O)CC4(CC4)C3)n21 39193,N1(C(CC(CC)C2CCC2)=O)CCC(C(=O)N(CCCN(C)C)C)C(C)(C)C1 39194,Cc1ccc(C=CC(N2CCCC(NC(=O)C=C3CCC(C)CC3)C2C)=O)nc1 39195,C1(C)(C(N(C)C(c2cc(C3CC3)no2)=O)=O)C=CCN1C(C1CC(CF)C1)=O 39196,c1(C(c2nnnn2CCOC(C)=O)OC)sc(Br)cc1NC(CC)C(=O)OC 39197,C1(C(=O)OC)CC(NCc2ccnc(O)c2)C12CCC2 39198,N1(C(C(CC)CC)=O)CCC2(CC1)CN(C(C1CCCC13CC3)=O)CC(C)O2 39199,C1(NC(C)C)CC(NC(C2COCCN2C)=O)C12CCC2 39200,C1(C(N2CC=CC(C(N(CCC)C)=O)C2)=O)CC(C)(C)CN1C 39201,c1(C(N(C)CC2CCCN2C(=O)C=CC2CCCO2)=O)cc(O)cc(C#N)c1 39202,C1(CNC(C=CC(=O)OCCCC)=O)CN(C(=O)CC)C2CCN1C2 39203,C1(CO)CCCC(N=c2[nH]c(=NC3CC(N4CCC4)C3)[nH]c3c2COC3)C1 39204,N1(C(=O)CC2CC(F)(F)C2)CCC2CCN(C(C3CC4CC3C4)=O)C2C1 39205,CC1CCC(NC(=O)CCC2(C#N)CCC2)CN1C(=O)CC1(N2CCCC2)CC1 39206,C1(C(N(CCCNC(c2ccc(F)o2)=O)CC)=O)CC1C1CC(F)(F)C1 39207,c1(C(=O)NCc2scc(CNC(CC3C(C)CCO3)=O)n2)cc(O)ncn1 39208,N1(C(c2ccc(SC)cc2)=O)CCN(C(=O)C=CC2CCCC2)C2(CC2)C1 39209,c1(OC)ccc(Cl)c(CC(=O)NC2CC(CCNC(=O)CCc3cc[nH]n3)C2)c1 39210,Cc1cc(=NCCCS(=O)(=O)C(F)F)[nH]c(NC2CCCOc3ccc(Br)cc32)n1 39211,N1(C(CS(N)(=O)=O)=O)CCC2CCCN(C(=O)Cc3cccc4[nH]ncc34)C2C1 39212,C1(C(=O)NCCN(C(C(N2CCOCC2)C)=O)C2CCCC2)CC(F)(CF)C1 39213,C(=O)(C(C)S(=O)(=O)C1CCOCC1)NC1C2CN(C(C(C)NC(CC)=O)=O)C1C2 39214,C(=O)(CCCC(CC)NC(c1cnn(C2CC2)c1)=O)N(C1CCOC1)CC#C 39215,c1(OC)noc(C2CC2)c1C(=O)NCC1CCCN1C(C1CC2CC2C1)=O 39216,c1(-c2cn(CC(COCC)(C)C)nn2)cc(C(=O)OC)ccc1NC(C)=O 39217,CCC(C)CCCC(=O)NCC(CNC(=O)Cc1cc(O)nnc1O)OC 39218,N1(C(C2CCCN(C(C3(C)ON=C(C)C3)=O)C2)=O)CCC2(CC1)CSC2 39219,c1(C(=O)NCC(CNC(CCC(C)OC)=O)OC)nn(C)c(C)c1[N+](=O)[O-] 39220,c1(C(=O)NCc2c(C(=O)NCCC(CC)CO)n[nH]c2)cccc2ccoc12 39221,C(=O)(CC1=Cc2ccccc2C1)N(CC(CC)NC(C1CC1C(F)(F)F)=O)C 39222,Cc1nc2cc(C(N3CCCC3CCCNC(=O)C(C)N(C)C)=O)ccc2s1 39223,C1(NCc2c(C)c(Br)ccn2)CCCC2CN(C(=O)OC(C)(C)C)CC12 39224,C1(CN(C(C(C)OC)=O)C)COCCN1C(=O)C(CO)OC 39225,C1(NC(C(n2cc(C3(C(N)=O)CC3)nn2)C)=O)C(C)(C)C(N(C)C)C1(C)C 39226,N1(C(C=CCCC=C(C)C)=O)CCC2(CCCN2C(=O)Cc2ncc(F)cn2)C1 39227,c1(C(N2CCCC2CC)C(=O)NC(CC)C)cnc(C2CC2C)s1 39228,C1(C(N(C2CCN(C(C3C(C)CCO3)=O)C2)C)=O)CCCN(C)C1 39229,CC1(C)CC(NC(=O)CC2C=CS(=O)(=O)C2)CN1C(=O)CCCn1ccnc1 39230,N1(C(C=C)=O)CC2(C1)CN(C(C1COCCN1C1CCCC1)=O)C2 39231,c1(-c2cn(C(NOCC(Cc3ccccc3)OC)=O)nn2)cc[nH]c(=N)c1 39232,c1(C(=O)NCC2C(NC(C=Cc3nnc(C(C)C)o3)=O)C2)nnc(O)cc1O 39233,C(=O)(CS(=O)(=O)c1ccccc1Cl)NCC1(O)CN(C(C(CC#C)O)=O)C1 39234,c1(C(N2CC(CCC)N(C(c3cncs3)=O)CC2)=O)ccc(Cl)c(F)c1O 39235,CC1(C)CN(C(=O)C=C2CCSCC2)CC1C(=O)NCc1ccccc1Cl 39236,C1(C(N(CC(C)CNC(c2sc(Cl)cc2Cl)=O)C)=O)CCCC1C1CC1 39237,C1(CNC(C2(SC)CC2)=O)CCC(C)CN1C(c1ccc(C2CC2)o1)=O 39238,c1(C(=O)NCC(CO)NC(C2CCC(C(=O)OC)O2)=O)cnc(C2CC2)nc1O 39239,C(CCN=c1nc(N2CCCC(F)(F)CC2)c2c([nH]1)CCC2)C1C(C)C1 39240,C(=O)(C(CC(C)C)N(C)C)NCC(C)NC(CC1C(C(=O)OCC)C1)=O 39241,N1(C(CCC#C)=O)CC2C(C(F)(F)F)CC2(NC(c2ccc(C)c(C)c2O)=O)C1 39242,N1(CCCN(C(=O)CCc2ccc(Cl)s2)C2CC2)CCCCCC1 39243,c1(OCC(=O)NCC(CO)NC(c2cnc(CC)[nH]2)=O)ccc(F)c(Br)c1 39244,N1(C(COCCCOC)=O)CC(C(=O)N(C2CCCC2)CCO)CCC1(C)C 39245,c1(C(=O)NCC2CN(C(=O)CCC3CCCC(O)C3)C2)cc(Cl)c(F)cc1Cl 39246,Cc1nc(C(C)(C)C)nc(S)c1C(=O)NCC1CC2CC2N1C(=O)C(C)C(C)C 39247,N1(C(C2OCC(=O)C2)=O)CCC(C2CCN(C(C3CN4CCN3CC4)=O)CC2)C1 39248,C1(CC(=O)NCCOCC(F)F)CCCCC1NC(C1(Cl)CCCCC1)=O 39249,C#CCC(C)(CC)C(=O)NCC1CN(C(c2ncsc2C2CC2)=O)CC1(C)C 39250,C1(N=c2[nH]n3cc(C)nc3s2)(CCC)CCN(C(C2CCCC(F)C2)=O)CC1 39251,N1(C(CC)=O)CCC2(CC1)C(NC(=O)Cc1ncn3c1COCC3)CS2(=O)=O 39252,CCCCCCCCCCNC(C1CC(Nc2cc(SC)ncn2)C1)=O 39253,CC1CC(C(=O)NC(C)(C)CCCNC(=O)Cc2cnc[nH]2)CCS1(=O)=O 39254,CC1CC(NC(C2(CF)CCC2)=O)CN(C(=O)CC2CCCCO2)C1 39255,CC(CF)CC(=O)N1CCCC(CN(C(=O)Cc2cccn2C)C)C1 39256,N1(C(c2nnc(C(C)(C)C)s2)=O)CC2(CC(NC(c3ncccc3F)=O)CO2)C1 39257,C1(NC(c2cccc(OC)c2)=O)CC(F)(F)CC1NC(c1scnc1Cl)=O 39258,c1(OC)ccnc(O)c1C(N1CC(CNC(=O)C=Cc2ccnn2C)C1)=O 39259,N1(C(=O)CC2CC2)CCN(C2CCCN(C(=O)C=Cc3cscn3)C2)CC1 39260,c1(OC)cnc(C(=O)N(C2CCCN(C(=O)C(C3CCCCC3)O)C2)C)c(F)c1 39261,N1(C(c2c(C(C)C)cnn2C)=O)CCCC2(C1)CN(C(=O)CC1=CCCCC1)C2 39262,C1(CN(CC)CC)(Cc2c(Br)ncn2C)CCN(C(=O)OC(C)(C)C)CC1 39263,C1(C(=O)NC(C(C)NC(C2CC3CC3C2)=O)CO)CC(C)(C)CO1 39264,C(c1cccc(C#N)c1)=NC(N1CCN(C)C(CO)C1)=O 39265,N#Cc1cccc(CCC(=O)Nc2nccc(F)c2F)c1 39266,C1(C(N(CC(C(C)C)OC)C)=O)C=CCN(C(C2CCC=CCC2)=O)C1 39267,C1(C(C(=O)N(C2CSC2)CC#C)C)CCN(C(=O)COC2CCCC2)C1 39268,CC(C)(CCNC(=O)CCc1ccon1)NC(c1coc(C(N)=O)c1)=O 39269,CC1CC(NC(=O)COC2CCCC2)CCN1C(=O)C=Cc1ccc(F)cc1 39270,C1(C(N2CC3C(CNC(CN4CCCC(CC)C4)=O)(C3)C2)=O)CC(C2CC2)=NO1 39271,c1(OC(C)(C)C)ccc2c(NC(N3CC(SCC(=O)O)C(O)C3)=O)cnn2c1 39272,C(C(C)(C)C(=O)NC1CCCN(C(=O)CCNc2ccccc2C)C1)SC 39273,n1(CC=C)cccc1C(=O)NC(C1CCN(C(C2(F)CC2)=O)C1)C 39274,C1(C(=O)NCCCCCCOC)CC2(CCC2)CN1C(C12CC(F)(C1)C2)=O 39275,C(=O)(C1=COCCO1)N(C)CCOCCCNC(c1ccc(C(C)(C)C)cn1)=O 39276,c1(C(N2C(C(=O)NCC3CC(=O)NC3)CC(F)C2)=O)nccc2ccccc12 39277,N1(C(C(C)OCCC=C)=O)CCN(C)C(CNC(C2CC(CC)(CC)C2)=O)C1 39278,C1(CC=C)(C(=O)NC(C=C)C2CCC2)CCCN1C(=O)C(C)CSC 39279,Nc1cncc(C(=O)NC2CCCCC2CNC(c2cc(Br)no2)=O)c1 39280,S(=O)(=O)(c1cccc(Cl)c1)N(CC(N1CCN(C(C(CC)OC)=O)C(C)C1)=O)C 39281,N1(C(C(C(C)C)OCC)=O)CC2(NC(=O)C(C)OC)CCC1CC2 39282,CC1CCCN1CC(=O)N(CC(=O)NC(c1cccnc1)CO)C1CCC1 39283,N1(C(c2ccc(OCC)nc2)=O)CCN(C(=O)CC2CC(N(C)C)C2)C(CC)C1 39284,C1(C(=O)NCC(C)NC(c2snc(OC)c2Br)=O)CCOC(=O)CC1 39285,N1(C(C(C=C=C)C)=O)CCCC(CCC)(NC(c2cc(Cl)ccc2Cl)=O)C1 39286,C1(OCC(=O)NCC2(NC(c3cc(C(F)F)no3)=O)CCC2)CCC(F)(F)CC1 39287,C1(C)(OC)CCCN(c2cc(NCc3nc(C)c(C)o3)nc(C(F)(F)F)n2)C1 39288,CC1CCN(C(c2n[nH]cc2Cl)=O)CCN1C(=O)CCCS(N)(=O)=O 39289,c1(N2CCC3(C(NC(c4cnco4)=O)CC3)CC2)ncc2c(Br)cccc2n1 39290,c1(NC(=O)CC2CC(NC(=O)Nc3cn[nH]c3)C2)ccc(-c2ccccn2)cc1 39291,c1(Cc2nc(-c3ccc(C(=O)O)s3)on2)cccc(F)c1 39292,C(=O)(C(C(C)(C)C)n1ccnn1)N(CC(C)O)CCNC(=O)COC1CCOC1 39293,C(=O)(CS(=O)(=O)CCO)N1CCC(C)(CNC(C2C(CC(C)C)C2)=O)CC1 39294,N1(C(C=C(c2n(C)ncc2)F)=O)CCCC2(CCN(C(=O)CN3CC=CC3)C2)C1 39295,C(=O)(C1=CCCCO1)NC(CCOC)C(=O)N1CC(C)=C(C)C1 39296,C1(C(=O)NCC2N(C(CN3C(C)CCC3)=O)CCC2)CC(S(C)(=O)=O)C1 39297,CC1CN(C(C2COC(C)(C)O2)=O)CC2(CCN(C(=O)CN3CCC3)C2)O1 39298,CC(C)CC(O)CC(=O)NCC(C)C(N1CCCC1(C)C1CC1)=O 39299,N1(C(c2cncc(OC)c2)=O)CCN(C(=O)CC(C)(F)F)C(C(C)C)C1 39300,C1(C)(NC(C(=O)N(C)Cc2ccc(-c3ccccc3)o2)=O)CCCC1O 39301,N1(C(c2[nH]c(CC)c(Cl)n2)=O)CCC(NC(c2ccn(CC(C)C)n2)=O)C(F)C1 39302,N1(C(C(=O)NCCC)CCCCCO)CCc2cc(C)cc(C)c2C1C 39303,N1(C(c2ccccc2)C(=O)Nc2cccc(F)c2)CCc2cc(F)cc(Cl)c2C1 39304,N1(C(=O)Cc2sccc2Cl)CCCC(N(CCO)C(C2CC(F)C(=O)N2)=O)C1 39305,CN1CCCC(NC(C2CC(=O)CN2C(=O)CC2CSC2)=O)CC1 39306,N1(C(C(c2ccn(C)n2)C)=O)CC=CCC1C(=O)N(C)CC1(C)CC1 39307,CC(C)CCCC(C)C(=O)NC1(C2CCCN2C(c2cnc(C(C)C)o2)=O)CC1 39308,N1(C(C2C(=C)C2)=O)CC2CC(CNC(c3ccc(C(C)(C)C)[nH]3)=O)C2C1 39309,C1(N(C(C)=O)C(C2CCN(Cc3nc(C(=O)O)co3)C2)=O)CCS(=O)(=O)C1 39310,C(=O)(C(C)(C)c1ccsc1)NC1(CCC(=O)NC2CC(N(C)C)C2)CCC1 39311,N(C1CCCn2ccnc21)C(C(CO)NC(C(C)n1cccc1)=O)=O 39312,n1(C(C)C)ncc(C(N2CCC(CF)(NC(=O)CC3CCCC(=O)N3)C2)=O)c1Cl 39313,N=c1ccn(CC(=O)NCC(C2CC2)NC(c2cnnn2C2CCOCC2)=O)[nH]1 39314,c1(C(N2CC(C)C(NC(c3c[nH]nc3-c3ccsc3)=O)C2)=O)cc(=O)cc(Cl)[nH]1 39315,c1(C(=O)NCC(C)(C2CCC2)NC(c2cc(C3CC3)ncn2)=O)ccc(F)cc1 39316,N1(C(C2(OCC)CCCC2)=O)CCCN(C(=O)Cn2nnc(=O)[nH]2)CC1 39317,C1(CCNC(C2C(OCC)C2C)=O)CCCN(C(c2ccc(F)c(Cl)c2)=O)CC1 39318,c1(C(=O)NCCC2CSCCN2C(=O)CC2COCCO2)cnn2ccsc12 39319,N1(C(c2c(C)cnc(F)c2)=O)CC(C)OC2(CCN(C(=O)C(=O)C(F)(F)F)C2)C1 39320,N1(C(C(C2CCCC2)OC)=O)CCC(NC(c2cc(C(C)C)on2)=O)CC(O)C1 39321,C(=O)(NNc1c(C#N)cccc1Cl)NCCc1cc(C)on1 39322,CC1CCCC(N2CCN(C(c3ccoc3)=O)CC2)C1 39323,c1(CCC(N2CCN(C(C3CC(=O)NC3)=O)CC2CO)=O)nc2ccccc2o1 39324,c1(C(=O)NCCC2N(C(C(C)OCC#C)=O)CCC2)ccc(OC(F)(F)F)cn1 39325,Cc1noc2ncnc(N3C4CCC3CC(NC(c3ncc(Cl)s3)=O)C4)c12 39326,c1(CN(C)C(C2(C)CC2)=O)cnn2c1CN(C(c1cc(F)ccc1F)=O)CC2 39327,C(=O)(C(O)C(F)(F)F)NC(C1CCN(C(C(COC)(C)OC)=O)CC1)CO 39328,C(=O)(C1=CCC(C)(C)CC1)N1C(CNC(c2cc(C(C)=O)sc2)=O)CCC(C)C1 39329,c1(OCC(=O)NC(CCNC(C2(C=C)CCC2)=O)C)ccc2c(c1)CCC2 39330,C1(C(=O)NCC(CC)NC(=O)C(c2ccc(F)cc2)(C)C)CCCCN1N=O 39331,C(=O)(C(Cn1ccnn1)NC(c1cc(C2CC2)[nH]n1)=O)NC(CCOCC)C 39332,c1(C(N2CCN(C(CC(C(CC)O)C)=O)CC2)=O)csc2cc(C)ccc12 39333,c1(C(N2CC(CCO)(NC(c3ccn(C4CCC4)n3)=O)C2)=O)ccc([N+](=O)[O-])o1 39334,C1(O)(CC(N2CC(O)(CCNC(C(C=C)(C)O)=O)C2)=O)CCN(C)CC1 39335,C1(C(=O)NC(C(C)C)(C)CNC(=O)CC2CC3(CC3)CO2)CC2(C1)CC1(CCC1)C2 39336,C(c1ccc(N(C)C)cc1)=CC(=O)NC(C(C)C)(C)CNC(c1n[nH]cc1F)=O 39337,C=C(C)CC(C(=O)N(CCC(=O)OCc1c(C)noc1CC)OC)OC 39338,N1(C(CCCC)=O)CCC(C)C(CNC(=O)CNC(=O)CC2CCCCC2)C1 39339,N1(C(CCCN(C(C2C(C(=O)OC)CC2)=O)C)=O)CCC12CCCCC2 39340,CCCCCCC(F)C(=O)N1CCC(C)(CNC(c2ccc(O)c(N)n2)=O)C1 39341,c1(C(=O)NCC(C)(C)OCC(=O)NC2CCC3(CC3)C2)cccc(CO)c1 39342,Cc1scc(C(=O)NC2CCCCC2CNC(c2cn(C)cn2)=O)c1N 39343,n1(CCNC(C2CCC(NC(C3CCSCC3)=O)CO2)=O)ccc2ccccc12 39344,c1(CC(=O)NC2CC(NC(c3c(COC)nn(C)c3)=O)C2)c(C)cccc1C 39345,C=CC1(CC(N2CC(CNC(C3(C)CCC3)=O)C3(CC3)C2)=O)CCOCC1 39346,Cc1cccc2c1CN(C(C1CN(C(C3C(C)C3C)=O)CCC1(C)C)=O)C2 39347,c1(N2CC(C)OC3(C2)CCC3)nc(NCC2C3COCC23)c2cnn(C)c2n1 39348,C1(C(=O)NCC(C)N(C(C(C(=O)OCC)CC)=O)C)CC2(C1)CC(F)(F)C2 39349,C=CCC(F)(F)C(=O)NCCC1(C)CCN(C(c2ccc(C3CC3)cn2)=O)CC1 39350,C(=O)C(CC(C)C)ONC(C1(C)CCSCC1)=O.c1(CNCC)ncc[nH]1 39351,C1(NC(c2c(OC)ccnc2)=O)CCCC2CN(C(C3(C)CCCC3C)=O)CC12 39352,n1(CCC(N2CCN(C(CSCCOC)=O)C(C)C2)=O)c(=O)oc2ccccc12 39353,c1(OC)nc(Br)ccc1NC(C1(F)CCN(C(c2ccccc2O)=O)C1)=O 39354,c1(C(c2n(CCC)nnn2)NCCCCOCC2CC2)cccc2nccn12 39355,Cc1cccc(OCC(N2CC(NC(C3(O)CCOCC3)=O)CCC2C)=O)c1C 39356,C(=O)(CCN=c1[nH]ccs1)NC1C(NC(C2C3CC(C)(C3)OC2)=O)CCCCC1 39357,n1(CC(=O)NC(C)CNC(=O)CN2CCCNS2(=O)=O)cc(S(N)(=O)=O)cn1 39358,N1(C(C2(OC)CC2)=O)CCN(C(=O)CSc2cccs2)C(c2ccccc2)C1 39359,C(C)(CO)(CS(C)(=O)=O)NCCCOCc1ccc(OC)cc1 39360,C(=O)(C(F)C(C)CNC(C1CC(=C2CCC2)C1)=O)NC(C(=O)NCC)(C)C 39361,C1(NC(C2(C#N)CCCC2)=O)CN(C(c2cnc(C3CC3)o2)=O)CCC1CO 39362,c1(OC)ncc(C(N2CC(C)(NC(C3CCC(OC)C3)=O)C2)=O)c(C(F)F)n1 39363,CC1(C)OCC2(CCN(C(c3coc(Cl)n3)C(=O)NC3COC3)C2)CO1 39364,C(=O)(CC1=CCCC1)NCC(=C)CCNC(=O)C(F)(F)c1ccccn1 39365,CC(C)S(=O)(=O)c1ccc(C(N2CC(NC(=O)C3=NNC(=O)CC3)C2)=O)cc1 39366,CC(C)CC(CC(=O)N(C)C(C1CCCCC1)C)NC(C1CC1CC(C)C)=O 39367,N1(C(CSCC(C)C)=O)CCC2CCN(C(C3CC4(C3)CC43CCC3)=O)CC12 39368,CCCC(CCC)CC(=O)N1CCCC1CNC(C1(CC)CC(C)(C)C1)=O 39369,c1(C(C)=O)ccc(C(=O)NC2CCC(CNC(c3ccc(Br)s3)=O)C2)o1 39370,C1(CNC(Cc2cc(C)[nH]n2)=O)COCCN(C(=O)Cc2ccccc2F)C1 39371,C1(NC(C(CC)OCC)=O)CN(C(c2cn(C(C)(C)C)nc2C)=O)CC12CC2 39372,C1(CNC(C(COC)O)=O)N(c2ccnc(C(C)(C)C)n2)CCCC1(C)C 39373,c1(C(N(CCC(C(C)C)NC(=O)CCOCC2CC2)C)=O)cccc(N)c1O 39374,CC1CN(C(c2ccc(C(F)(F)F)[nH]2)=O)CC1CNC(C1(S(C)(=O)=O)CC1)=O 39375,N1(C(CC2CC(C)C2)=O)CC(CNC(c2ccc([N+](=O)[O-])s2)=O)C(C)(C)C1 39376,C1(=CC(=O)NC2(CNC(Cc3cn(CC)nc3)=O)CC2)CCCCCC1(F)F 39377,C1(CNC(C2(CCC)CC2)=O)CCC(C)CN1C(c1cc(C(F)F)ccc1Cl)=O 39378,c1(CC)ccc(F)cc1C(N1CCC(NC(=O)CSC(F)F)C(CC)C1)=O 39379,n1(CCC)nc(C)cc1C(=O)NCC1CC1CC1CC1.C12CC1CC2=O 39380,N1(C(c2ccc(N(C)C)cc2)=O)CCC2(CCC(NC(=O)OC(C)(C)C)CC2)C1 39381,C12C=CC(C1)CCOC(=O)N2.N1(CNC(=O)C(=O)NC(C)(C)C)CCOC1=O 39382,C1(C(N(CCC(F)(F)F)C)=O)CCC(C)(C)N(C(c2csc(=N)[nH]2)=O)C1 39383,c1(C(N(CCC(C)NC(=O)CC(C)c2cccnc2)C)=O)ncncc1Cl 39384,CCCCS(=O)(=O)NC(C)C(N1CCC(CNC(C2CCCCC2C)=O)CC1)=O 39385,c1(OCC=C)ccc(Cl)nc1C(N1CCC(C(C)CNC(=O)CCOC)CC1)=O 39386,N1(CCCNC(CC2(C)CCCC2)=O)CCN(C(=O)CCC(F)F)CC1 39387,N1(C(C2(CC=C)CCC2)=O)CCC2(C1)CN(C(=O)C(C)NC(=O)OC)CCO2 39388,C1(NC(C2CCC(CC)CC2)=O)C2CC3C1C3C2C(=O)N(C1CCCC1C#N)C 39389,C1(N(C)C)CC(N=c2[nH]c(=NCCP(C)(C)=O)[nH]c3c2CCCC3)C1 39390,N1(C(c2ccc(CC)o2)=O)CC=C(CCNC(=O)C(C)COc2ccccc2)CC1 39391,C(=O)(C(CC)CC=C)NC1(CC=C)CN(C(C2(Cc3cnn[nH]3)CCC2)=O)C1 39392,n1(CC)ccc(C(N2CCC(CNC(=O)CCc3cncs3)C23CC3)=O)cc1=O 39393,CCCCC(C(=O)N=c1ccn(Cc2ccc(C(F)(F)F)cc2)[nH]1)C(C)C 39394,C1(C#N)(C(=O)NCC(CNC(c2ccc(N(C)C)cc2)=O)F)CCS(=O)(=O)CC1 39395,CCC(C)CC(C(=O)N(CC(N)=O)C)NC(=O)CCCC(F)(F)F 39396,C1(NC(CC2CCN(C(C(CC)(C)O)=O)CC2)=O)CC12CCCCCC2 39397,C1(CC(=O)NCC(C)(C)OCCNC(CC(=O)NCC)=O)CCCCC1C 39398,C=CCC(CC(C)C)C(=O)NC(C1CCCN1C(=O)C1=CCCS1)C 39399,c1(C(=O)NCC2(CNC(c3c(C)scn3)=O)CC2)cnn(C2CCOCC2)c1C 39400,C1(C(=O)NCCCCC#C)(OC)CCN(C(c2cc(C)cc(F)c2)=O)CC1 39401,C(CC(O)C(=O)NC1CCOCC1F)NC(C1N(C(C)C)CCC1)=O 39402,N1(C(c2c(CC)nc(C)[nH]2)=O)CC2(CCN(C(=O)CCCCF)C2)C1 39403,C(=O)(CCCCC(C)C)NC(CCN(C(C=Cc1n(CC)ncc1)=O)C)C(C)C 39404,C1(C(=O)NCC(C)(C)NC(=O)CCc2ccc(C#N)cc2)CCS(=O)(=O)C1(C)C 39405,C1(CNC(c2c(CC)scc2)=O)COC(C(F)(F)F)CN1C(C1CC(F)(F)C1)=O 39406,c1(C(N2CCCC(CN(C)C)C2)=O)ccc(N=[N+]=[N-])cc1 39407,c1(C(=O)NC2(C)CCCN(C(C(CC(C)C)(C)O)=O)C2)ccnc2c1CC(=O)N2 39408,N1(C(CC(C(C)C)NC(c2c(C#C)cnn2C)=O)=O)CCC2(C=CCO2)C1 39409,N1(C(c2c(CC)ocn2)=O)CCCCC1CCC(C)(C)NC(c1occc1C)=O 39410,c1(OC)cc(CNC(CN2CCCC(C(=O)N(C)C)C2)=O)ccc1O 39411,O=C(C#CC1CCCOC1)NCC1CN(C(=O)Cc2ccc(Cl)cn2)C1 39412,C1(CCNC(=O)C(C2CCCCC2)F)CCCN(C(=O)Cc2cccnc2)C1 39413,c12cccc3cc(oc13)N2S(=O)(=O)CCC1CCOCC1.N1(CC)CCCCC1 39414,CC1CCCCC1(C)NC(=O)C(c1cnn(C)c1)NC(=O)CC(=O)NC1CC1 39415,C(=O)(C(CCCO)c1ccccc1)N(C(C)C)CCN(C(=O)COCC(F)F)C 39416,C1(C(N(CC)CC2CCC2)=O)CCCC1CNC(=O)CCCn1ccnn1 39417,C1(C(CC)C)CCN(C(C2CCC2NC(c2ccc(=N)[nH]c2)=O)=O)CC1 39418,c1(C(=O)NC2CCCC(NC(C(CCSC)O)=O)C2)nccc2nn[nH]c12 39419,CCC(CC(=O)N1CC2CCN(C(=O)Cc3cnccn3)C(C2)C1)CC(F)(F)F 39420,C(c1ccc(C)c(Cl)c1)=CC(=O)NC1C(NC(C(n2ccc(C)n2)C)=O)C1 39421,c1(COCCC)cn(C2CC3(C(=O)N(C(C)C(=O)OC)C4CC4)CC23)nn1 39422,c1(C(c2nnnn2C2CC(F)(F)C2)NC2CC(CC)C2)cncn1C1CC1 39423,C(C(COC)C(=O)N1CSCC1C(=O)NCCn1cnnn1)OC 39424,N1(C(c2ccc(OC)nc2)C(=O)NCCCC2CC2)CCC(O)CC1C 39425,c1(C(N2C(COC)(CNC(C3CC(C)CO3)=O)CCC2)=O)ccc([N+](=O)[O-])n1C 39426,C(C(C)(O)C(=O)N(CC(C)N(C(=O)CCn1cncn1)C)C)OC 39427,CC(O)C(C)C(=O)N1CCN(C2CCN(C(C34CC3C4)=O)C2)CC1 39428,c1(OCC=C)ccccc1C(=O)NCCC(C)CCNC(c1cc(Cl)n(C)n1)=O 39429,N1(C(C2C(C)C2C)=O)CC(CNC(=O)CC2CC(C)OC2C)OC(C)(C)C1 39430,N1(c2c3ncn(C(CC)(C)CC(C)O)c3ncn2)CCCn2cc(Br)cc2C1 39431,c1(C(C)=O)ccc(C(C)NC(=O)C(N)Cc2ccc(F)cc2)cc1C 39432,N1(C(CONC(C#CC(C)C)=O)=O)CCC(C2CCOC2)C1 39433,N1(C(CCOCC#C)=O)CC(CNC(=O)C(CO)c2ccccc2)CC12CCC2 39434,c1(C(N2CCSCC2C2CCC2)C(=O)NCCCF)cc2c(Cl)nccc2s1 39435,C1(CCCNC(CCOC)=O)CCCCN1C(=O)C(N1CCC(C)CC1)=O 39436,C1(C(N2CCC(=CCNC(c3c(CC)nns3)=O)CC2)=O)CN(CP(C)(C)=O)C1 39437,C1(CNC(C2(C(N)=O)CCC2)=O)CCN(C(c2cnn[nH]2)=O)C12CCC2 39438,N1(C(CCSC)=O)CCCC1C1CCCCN1C(=O)CN(C)CCO 39439,c1(N2CC3CC(NC(c4ccc(C)o4)=O)C3C2)c(Cl)cccc1[N+](=O)[O-] 39440,c1(CN(C)Cc2onc(C(C)OC)n2)cc(OC)c2c(c1)OCCO2 39441,CC(C)CCCCCC(=O)N(C)CC1(O)CCN(C(=O)CCC#N)CC1 39442,C1(C(N2CCC(CNC(CCn3ncc(C)c3)=O)C2)=O)CCC(C(C)C)CC1 39443,c1(C(C(=O)NCC2CC2)N(C2CCN(C(C#C)(C)C)CC2)C)cc2n(n1)CCCC2 39444,c1(C(CC(=O)OC)NC(=O)CNC(N)=O)cccc(-c2cccnc2)c1 39445,CCC(C)CCC(=O)NCC(c1ccc(F)cc1)NC(=O)C=Cc1cc[nH]c1 39446,C1(NC(COCC#C)=O)CCOC(CNC(=O)CC2COCC2(C)C)C1 39447,C1(Cl)(C(=O)OC)CC1C(=O)NCCC(C)NC(C1(N(C)C)CC1)=O 39448,C1(CCC)CN(C(=O)C(C)CSC)CC1NC(c1ccc(C)nn1)=O 39449,N#CC1CCCC1NC(C1CCCCN1c1ncccn1)=O 39450,C1(NC(C=CC(CC)C)=O)CCCCCN(C(=O)Cc2ccsc2)C1 39451,C(=O)(C(C)(C)C(F)(F)F)N1CC(c2cn(CCC=C=C)nn2)C(C)(C)C1 39452,C(C(C)(C)C(c1nnnn1C(C)C(=O)OC)NCc1sccc1C)OCC 39453,c1(CCC(=O)NC2C(NC(CCCNC(C)=O)=O)CCC2)cccc(F)c1F 39454,c1(CCC(=O)NCC(CNC(=O)C(C)C#N)OC)ccc(C(C)C)cc1 39455,CC(C(=O)N1CC(NC(=O)C(n2cc([N+](=O)[O-])cn2)(C)C)C1)C(C)(C)C 39456,Cc1ccc(F)cc1N(C(=O)C(C)NC(c1cc(Cl)cs1)=O)C 39457,Cc1cc(F)cnc1C(N1CC(NC(=O)C(c2cccc(Cl)c2)O)CC(O)C1)=O 39458,c1(-c2nc(NC(=O)NC3COC4(CCCCC4)C3)sc2)cnc2ccccn2c1=O 39459,c1(C(=O)NCC2CN(C(C3C(C)(CC)C3)=O)C2)cnn(C(F)(F)F)c1 39460,c1(C(=O)NC2CCCC(NC(CN(C)C(N)=O)=O)C2)n[nH]c2c1CCSC2 39461,O=C(CCc1cscn1)NNC(=O)N1CC(Cn2cc(COC(=N)O)nn2)C1 39462,C1(N(C(c2ncnn2C)C)CC2CC2)CCC12CCN(C(=O)OC(C)(C)C)CC2 39463,CCC(CCC(=O)N1CC=C(C)CC1)NC(=O)CCNC(=O)NC 39464,N(C(=NCCC(=O)NC(C)C)NCC1CCSC1)CC(CC)(C)C 39465,c1(C(OC)CC2CCCC2NC(c2sccc2-c2cccs2)=O)cn(CC)nn1 39466,CCC(C)(C(=O)NC(C1CCN(C(=O)C(C)(C)c2ccccn2)CC1)C)OC 39467,C1(C(=O)NC(C#CCC)(C)C)CCN(C(=O)C(=O)C2CCCCC2)O1 39468,C1(OC)CC(NC(C2CC(O)C2)=O)CN(C(c2cc(C)oc2C(F)(F)F)=O)C1 39469,c1(OC)ccc(Cl)cc1C(N1CCC(CCNC(C2(C)CCN(C)CC2)=O)C1)=O 39470,C(=O)(C(C)(O)C(F)(F)F)N1CC(CNC(=O)CCn2cccn2)CC(C)C1 39471,N1(c2nc(N3CC(C)CC(C)C3)nc3c2SCC3)CCc2nc(O)nc(O)c2C1 39472,c1(SC)ncc(C(N2CCSC(C(=O)Nc3ccc(Br)nc3)C2)=O)c(Cl)n1 39473,C(c1ccsc1)=CC(=O)NC(C)CCN(C(=O)C(C)N1CCCC1)C 39474,Cc1noc(C2CC2)c1C(=O)NC(CNC(c1ccnc(C2CC2)c1)=O)C(C)C 39475,CC(C(C)NC(=O)CSc1nncs1)NC(c1csnn1)=O 39476,c1(CCN(C(=O)NC2CC2C(=O)OC(C)(C)C)C(=O)OC)ccc(Cl)c(C)c1.CN 39477,C1(C)(C(N2CCC(OC)CC2)=O)CCCN(c2nccc(C(=O)O)n2)C1 39478,c1(NCCCNC(C(CCCC)O)=O)ncnc2sc(COC)cc12 39479,N#CC1CCCC(C(N2CCN(CC(=O)NCc3cnccn3)CC2)=O)C1 39480,C1(CCC)CCCN1CC1CC1CO 39481,C(=O)(C(CC(C)(C)C)NC(=O)C(CN(C)C)N(C)C)NCCCOCCCC 39482,C1(C(C)NC(CCCOCC=C)=O)CCCCN1C(=O)CCc1nccn1C 39483,c1(C(=O)NC(C(C)NC(COC(CC)CC)=O)C)cc(C)c(F)cn1 39484,c1(N(CC#C)C(c2cccc(N3CCCC3=O)c2)=O)cccnc1OC(C)C 39485,c1(C(N2CCC(CS(=O)C)C2)c2ccc(C(F)(F)F)o2)ccc2ncnn2c1 39486,C(=O)(CCCC)NC(C1CCN(C(=O)C(F)(F)c2ccccc2)C1)(C)C 39487,Cn1cc(C(N2CCCC2Cl)=O)c(C2CCC2)n1 39488,c1(CC)cc(=NC(=O)C2CC(C)(C)CCN2C(c2cccc(=O)n2C)=O)[nH]n1C 39489,C(=O)(C(CC)CC(F)F)NCC(CCOC)NC(c1n(C=C)ncc1)=O 39490,CN=c1[nH]cc(C(=O)NC2(C(=O)NC(C34CC(CO3)C4)C)CCCC2)s1 39491,N1(C(C(CCOCC)NC(CCC#CC)=O)=O)CC(CC)CC(C)C1 39492,CCCCC(O)C(=O)NCCc1cc(C(N2CCCC(C)C2CO)=O)no1 39493,C1(C(=O)NCCc2n(C)c(=O)on2)C2CC3C(C2NC(=O)CC2CCC(=O)C2)C13 39494,C1(CC(=O)N(C(CC)C(=O)NCCC2(C)CC2)C)NC(=O)NC1=O 39495,c1(C(=O)NC(C2CCCN(C(=O)COC(F)(F)F)C2)C)ccnc2ccccc12 39496,C1(NC(c2cnc(CC)[nH]2)=O)CCN(C(c2nc(Br)cnc2N)=O)CC1C 39497,CC1(C)CCCC1NC(=O)C(N1CCCC(C)C1)=O.c1(N)nc(C(F)(F)F)cs1 39498,c1(C(=O)NCCC2(NC(C3CC3(F)Cl)=O)CC2)c[nH]c2ccncc2c1=O 39499,N1(C(c2cc(COC)no2)=O)CC(F)CC1CC(N1CCC(O)(C(F)F)C1)=O 39500,N1(Cc2ccc(C)cc2)CC2CN(C(=O)NNC(=O)C(C)C)CC2C1 39501,N1(C(c2c(C)c[nH]n2)=O)CCCC2CN(C(=O)Cc3ccc(C#N)cc3)CC12 39502,Cc1cc2ccccc2cc1C(=O)NCC(O)CNC(c1cc(Cl)ccc1N)=O 39503,Cc1nc(CNC(c2nnsc2N)=O)oc1C(=O)N(C)CCOCCCO 39504,C=CC(C)(O)C(=O)NC(C)CCNC(=O)CCn1ccc(=N)[nH]1 39505,c1(C(=O)NCC(C)CC(F)F)n[nH]c2cc([N+](=O)[O-])ccc12 39506,Cc1cccc2c1CCN2C(=O)CC(CC1CC1)NC(=O)COCCN(C)C 39507,Cc1ccc(C(=O)NCCNc2ccc(Nc3ncc(Br)cn3)cc2)cn1 39508,[SH](=O)(=O)c1ncc(F)cn1.CC(CS(C)(=O)=O)C(C)c1ccc(C)o1 39509,c1(C(C)C)noc(C(c2nnnn2C2CCCC2)NCc2cnn(C)n2)n1 39510,C(C)(C)(C(C)NC(=O)CCCc1cc(C)no1)NC(CSCCC)=O 39511,C1(CNC(c2nc(-c3ccccc3)ns2)=O)CCC12CC(F)(F)C2 39512,c1(OC)c(C(N2CCC(O)(CNC(=O)C(C)OC)C2)=O)csc1C 39513,N1(C(C2CC(C#N)C2)=O)CCC(O)(CCNC(C2CC(=O)N(C(C)(C)C)C2)=O)C1 39514,c1(NC(C2(C)CN(c3ncncc3Br)C2)=O)cc(C#N)cn1C(C)(C)C 39515,Cc1ccc2nc(N3CC4CC3(CNC(=O)CC3C=CS(=O)(=O)C3)C4)sc2n1 39516,N1(C(CNC(Cn2c(C)cc(C(=O)OC)c2C)=O)=O)CCCC2CNCC12 39517,Cc1cc(C(F)(F)F)c2cc(C(=O)NC(C)CCN(C)C)oc2n1 39518,CCC(CC)C(O)CNC(=O)CC1CN(C(=O)CCc2ccco2)CC1C 39519,N1(C(C=CSC)=O)CC(N(C)C(c2cccc(-c3ccco3)c2)=O)C(C)(C)C1 39520,N1(S(CC)(=O)=O)CC2CCCN(C(c3nccnc3C(N)=O)=O)C2C1 39521,CON(C)C1CN(C(=O)CC2CN(C(=O)C(C)(C)C3CCOC3)CCC2C)C1 39522,c1(N(CCCCO)C)nc(=NCc2cc(F)ccc2Cl)[nH]c2c1COCC2 39523,CS(=O)(=O)c1cc(C(N2CC3CC(C2)N(C(=O)C=C(Cl)Cl)C3)=O)co1 39524,C1(C(=O)NC2(CCC)CCC2)CCCN(C(C2CCC(OC)C2)=O)C1C 39525,C1(SC)CCC(N=c2nc(N(C)CC3CCCC3O)c3c([nH]2)CCOC3)CC1 39526,C(=O)(C(F)(F)C(O)C1CC1)N1CCC(N(C(C(C(C)C)NC(N)=O)=O)C)CC1 39527,c1(C(OC)OC)ccc(C(N2CCC(NC(=O)Cc3nccn3C)C2)=O)o1 39528,c1(OCC)cc(C(=O)NCC(C(C)C)NC(c2cocc2C)=O)ccc1OC 39529,N1(C(=O)OC(C)(C)C)CCN(C(c2cccc3oncc23)=O)CCCC1C(=O)O 39530,CC1CC(=O)CCC1C(=O)NCC=CC(=O)N(CCN1CCCCC1)C1CC1 39531,N(C)(S(N)(=O)=O)CC(=O)N(C1CC(NC(=O)CNC(c2ccco2)=O)C1)C 39532,C(=O)(C(CC1CCCO1)C(F)(F)F)N1CC(CNC(c2csnc2Cl)=O)C1 39533,CC(CS(C)(=O)=O)C(=O)NCC#CCNC(=O)CCC(=O)NC1CCCC1 39534,C1(NC(COCC(=C)C)=O)(CO)CCN(C(c2ccc(CO)s2)=O)C1 39535,CC1(C(=O)NC2CCC(CNC(=O)CSc3nncs3)CC2)Cc2ccccc2N1 39536,c1(CC)ccc(C(N2CCCC2CN(C(=O)Cc2cc(C3CC3)no2)C)=O)o1 39537,CN1CCn2ncc(C(N3CCC4CN(C(=O)COc5ccon5)C4C3)=O)c2C1 39538,c1(C(N2CCC3(C(C(=O)Nc4cnoc4)C3)CC2)=O)cc(F)c(Br)cc1[N+](=O)[O-] 39539,c1(C(N2CCC(NC(C(CC#C)(C)C)=O)C2)=O)cc2c(C)[nH]nc2s1 39540,c1(C(N2CC(CNC(CCSC)=O)C2)=O)ccncc1Cl 39541,C(=O)(C(O)CC(F)(F)F)NCCC1CCC(NC(C2CC3(CC(OC)C3)C2)=O)C1 39542,CCCC(C)(C)C(=O)NCC1CCC(C(N2CCC(CCOC)C2)=O)CC1 39543,C1(C)(C(=O)NC)CCN(C(=O)C(=O)Nc2cnn(-c3nccs3)c2)CC1 39544,c1(COC)nc(=N)[nH]cc1C(N1CC(NC(=O)C(O)C2CC2)C1)=O 39545,C1(NC(c2c(C)con2)=O)CC2(C(=O)NC3CC(CO)(CO)C3)COC1C2 39546,C12(C(=O)NC(C3CN(C(C4CCCC(C)(C)C4)=O)C3)C)CC=CCN1CCC2 39547,C1(C(=O)NC2CCN(C(c3nccc(SC)n3)=O)CC2F)Cc2ccccc2C1 39548,C1(C(=O)NCC23C(CN(C(CCC(N)=O)=O)C2)CCO3)CCCCC12OCCO2 39549,Cc1ccn2nc(C(N3CC4CCC3C4NC(c3nncs3)=O)=O)nc2n1 39550,c1(CC)cc(C(=O)NC2(CO)CN(C(C3CCCC3O)=O)C2)sc1C 39551,C(=O)(CC(C)CNC(C1CC(O)CN1C(=O)CP(C)(C)=O)=O)OC 39552,c1(CNC(=O)NC(c2ccc(OC)c(F)c2)C)c(C)cc(Cl)nc1Cl 39553,c1(OC)c(F)cc(C(=O)NCC2CCN(C(=O)CCCSC)CC2)cc1Cl 39554,N1(C(CCCOC)=O)CCC2CCCC12CNC(c1cc(Cl)ccc1F)=O 39555,C(=O)(N=c1nc[nH]n2cccc12)C1C2(CN(C(c3ccc(C#N)cc3Cl)=O)C2)C1 39556,C(=O)(C(F)C(C)(C)O)NC1CC(C(C)NC(c2cncc(CC)c2)=O)C1 39557,C(=O)(C1CCCc2n[nH]cc21)N1C2C(NC(=O)CCn3cnnn3)(CCC2)CC1 39558,C1(CNC(CS(CC)=O)=O)(NC(=O)C(C)Oc2ccccn2)CCC(C)(C)CC1 39559,C1(CC(=O)NC2(C)CN(C(C(C)n3ccnc3)=O)C2)CCCC(C)(C)CC1 39560,c1(CN(C2CCCC23CCNCC3)C(COC)=O)c(O)c(Cl)cc(Cl)c1Cl 39561,C(=O)(NNc1cc(C(F)(F)F)ccc1F)c1cnc2ccn(C)c2c1 39562,N1(C(c2ccc[nH]2)=O)CCC(N2CCN(c3ccc(F)cc3)CC2)CC1 39563,N1(C(=O)CC2(C)CC2(F)Cl)CC2CCCC1C2C(=O)NCC(OC(F)(F)F)C 39564,CC1(C)OC(=O)CC1C(=O)NC1(CC(=O)NCC2(C)CCCS2)CC1 39565,Cc1cn(CC(N2CCCC2CNC(c2ccsc2)=O)=O)c2ccccc12 39566,Cc1ncc(Cl)cc1C(=O)NCC1(C(F)F)CCN(C(=O)C(C)N2CCC2)C1 39567,N1(C(C2CC23CCC3)C(=O)NCCCOC)CC(C)OCC(C)(C)C1 39568,C1(C2CCC2)(C(N2CC(CC)N(C(C3CC4(CCCC4)C3)=O)CC2)=O)CC1(F)F 39569,N1(C(N(CC(O)CN2CCCC2=O)C)=O)CCCCCC(S(C)(=O)=O)C1 39570,N1(C(C2C(C)(C)CC2)=O)CCC2C1CCCN2C(=O)COc1cccnc1 39571,c1(C(=O)NC(C(C)NC(c2cc(CC(C)C)on2)=O)C)cc2n(n1)CCC2 39572,c1(C2(C(=O)OC)CCC2)cc(NCC(O)CNC(C)=O)ncn1 39573,C1(C(N2CC(CCNC(CN(C(C)=O)C)=O)OCC2)=O)CC2(C1)CC2(F)F 39574,C1(NC(CCSC)=O)C2CN(C(=O)CCn3cccnc3=O)CC12 39575,C=CC(CCC)CC(=O)N(CCNC(C1CCN(c2nc(C)cs2)CC1)=O)CC 39576,C(=O)(CC(F)(F)CC(=O)NCC1CCN(C(C2C=CCCC2)=O)C1)OC 39577,C1(C(=O)NCC(C)N(C(=O)C(C2CCOC2)OC)C)(CC)CCOCC1 39578,C1(CCCNC(C2C(Cl)(Cl)C23CC3)=O)CCCCN1C(=O)Cn1nccn1 39579,N1(C(C2C(C=C)CC2)=O)CCN(C(c2cnn(C(C)(C)C)c2)=O)C(CO)C1 39580,N1(C(CCN(C(C(CC(C)(C)C)OC)=O)C2CC2)=O)CCN2CC(F)CC2C1 39581,Cc1cc(C(F)(F)C(=O)NC2CC(CNC(c3cc[nH]c3C3CC3)=O)C2)cs1 39582,c1(C(C(=O)NCC(C)(CO)NC(=O)CNC=O)O)ccc(F)cc1Br 39583,CCC(CC)C(C(=O)N1CC(NC(=O)CC2CC2)C(CO)C1)OC 39584,CCC(O)C(C)C(=O)N(C)CC1CCCCN1C(=O)C(CCC)NC(N)=O 39585,C1(CNC(C2(C=C)CCC2)=O)(NC(=O)C=Cc2cncn2C)CCCCCC1 39586,n1(CC)ccc(C(=O)NCC(CO)NC(c2c(C)coc2C(C)C)=O)c1C 39587,Cc1nc(O)[nH]c1C(=O)NCCC1CCN(C(c2ncoc2C2CC2)=O)CC1 39588,C1(SC)CN(C(=O)CCn2cc(Cl)cn2)CC1NC(C1CCN(C)C1)=O 39589,C(C)(N=c1[nH]c(=NCc2ccc(N)cc2F)[nH]c2c1COC2)c1ccc(C)cn1 39590,c1(NC(C2CCCC(NC(C(C=C)(F)F)=O)C2)=O)cccc(F)c1C 39591,CC1CCOC(C(=O)N(C(C(F)(F)F)C2CC2)C)C1 39592,c1(C(=O)NC(CN(C(c2c[nH]c3nccc-3c2)=O)CC)C)sc2cncn2c1C 39593,c1(C(=O)NCC2(NC(CCCOC)=O)CCCCC2C)cnc2c(c1)COCC2 39594,N1(C(=O)NC(c2c(CCC)nns2)C)CCC(CO)C(O)CC1 39595,c1(C(N2CCC(CCNC(C3CC(SC)C3)=O)CC2)=O)c(F)cncc1Cl 39596,N1(C(c2cc(OCC)n[nH]2)=O)CCC2CN(C(=O)C(C)(C)C)CCC2C1 39597,c1(NC(CNC(C2(CC#C)CC=CCC2)=O)C2CC2)ncn(C)c(=O)c1Br 39598,c1(C(=O)NCC(C2CC2)NC(c2cc(C3CC3)no2)=O)ccc(Cl)cc1 39599,C1(C(=O)NCC(=O)OCC=C)CCN(C(=O)C(CC)SC)CCO1 39600,C1(CNC(c2n(C)cnc2)=O)CCCN(C(=O)Cc2ccn(CCF)n2)CC1 39601,C(CCCCC(=O)NCC1(C(=O)NCC2COC(C)(C)C2)CC1)=CC(C)C 39602,C(=O)(CCCC(=O)N(C)C)N(CCC(=O)NC(C(=O)NCC)C)C1CC1 39603,C1(C)(C(=O)NCc2cccc(CN(C(COCCOC)=O)C)c2)CCCS1(=O)=O 39604,C1(C(=O)NCC2(C)CCCN(C(CC3(C)OCCO3)=O)C2)OCCOC12CCC2 39605,c1(N(CC)CC)ccc(C(N2CCN(C(=O)NC3CC(=O)C3(C)C)CC2)=O)cc1 39606,Cc1cc(C)n2ncc(C(N3CCOCC(N4CCCC4)C3)=O)c2n1 39607,c1(C(=O)NCC2(F)CCCN(C(c3n(CC)ncc3)=O)C2)ccc2[nH]ccc2n1 39608,N(C1CC(C)(C)CCc2ccccc21)C(NNc1ccc(C)cc1Br)=O 39609,N1(C(C(CC)O)=O)CCN(C(=O)Cc2cncc(F)c2)C(CC)C1 39610,Cc1cc(C(=O)NCC2(C)CCN(C(=O)C(C)(C)O)CC2)ccc1I 39611,CCCC(C(=O)N1CCC(NC(=O)CCc2cnc(C3CCC3)o2)C1)C(C)C 39612,c1(C(N2CCCC(N(C(CC3N(C)CCC3)=O)C)CC2)=O)ccn2ccccc12 39613,N1(C(CC(c2ccc(C)cc2)(C)C)=O)CC(NC(c2ccc[nH]2)=O)CC(C)(C)C1 39614,C(C(C)CC(=O)NCc1ccc(CCn2cccn2)o1)NC(=O)OC(C)(C)C 39615,c1(OCC(=O)NCCCN(C(C(CC=C)C)=O)C)ccc(F)cc1F 39616,Cn1c(I)cc2c(N(C(c3cnnc(Cl)c3)=O)CC3(O)CNC3)ncnc12 39617,N1(C(c2cccc(NC)n2)=O)CCCC12CCN(C(=O)CN1CCC1C)CC2 39618,C1(CC)CCN(C(=S)Nc2ccc(OC(F)(F)F)cc2)C1 39619,C12(C(=O)NCCOCCCNC(c3c(C)nc(C4CC4)[nH]3)=O)COC(CCO1)C2 39620,c1(CC(=O)NC2(CO)CCN(C(C=Cc3cn(C)nc3)=O)C2)cc(F)cc(Cl)c1 39621,CC1CC(CCNC(c2cnn(C)n2)=O)CCN1C(=O)CCNC(=O)C=CCl 39622,C(CCN(C(=O)CCCOc1cccc(Cl)c1)C)(C(C)C)NC(C1(OC)CC1)=O 39623,c1(OC)cc(C(=O)NC(C2CN(C(C3C4CC5C(C4)C35)=O)CCO2)C)ccn1 39624,N1(C(C(CC)O)=O)CC(C2CN(C(c3ccc(C)c(O)c3)=O)C2)C1 39625,C1(C(N)=O)(CNC(c2cnc(-c3ccccc3)[nH]2)=O)CN(C(C2OCCO2)=O)C1 39626,C(=O)(C(C)(O)CCc1ccccc1)NCC(CO)NC(CCCN(C)C)=O 39627,c1(CNC(c2c(C(=O)OC)ocn2)(C)C)ccc(Br)cc1Cl 39628,C1(NC(CCC#C)=O)CC(CNC(=O)CCc2nc(-c3ccoc3)no2)C(O)C1 39629,N1(C(C2C(OCC)C2)=O)CCC(F)(F)C(CNC(=O)Nc2ccc(Cl)nc2OC)C1 39630,N1(C(CC2CCC(C)(C)O2)=O)CCCC(CC(=O)NC2COCC(C)(C)C2)CC1 39631,C1(C(=O)NC2CCC(NC(C(CC)OCC)=O)CC2)CCC2CC2CC1 39632,c1(OC)ccc(C(=O)NCCCC(C)(C)NC(c2onc(OC)c2Br)=O)cc1 39633,C1(C(=O)NC2CN(c3ncco3)C2)CCCCN(C(=O)C2CC2)C1 39634,N1(C(C2C(C)(Br)C2)=O)Cc2ccccc2CC1CNC(C1CC(F)(F)C1)=O 39635,N1(C(C(C2CCN(C(C3(C4CC4)CC3)=O)C2)C)=O)CCC2CN(C)CC2C1 39636,c1(CC)ncc(Cl)c(C(N2CCCCC2CNC(c2nc(C)ccc2C)=O)=O)n1 39637,Cc1nc2ccccn2c1C(=O)NC1COCC1NC(=O)CCC(C)(F)F 39638,C1(NC(C2(C(C)(C)OC)CC2)=O)CC2CC1N(C(C1(C(F)F)CCCO1)=O)C2 39639,CC(C)(CCCCNC(C1CC=CC(O)C1)=O)NC(=O)CC1CC1C1CC1 39640,C(=O)(C(CCSC)N(C)C)NCCOCCN(C(CC(C)N1CCCC1=O)=O)C 39641,c1(OC)ccc(-c2cn(CC3CCN(C(C4CCCCO4)=O)CC3)nn2)cc1F 39642,CC1(C(=O)NCC2CC(O)CN2C(C2COCCN2C=O)=O)CCCNC1=O 39643,N1(C(CCC(=O)OC)=O)CCC(C)C(NC(C2CN(C(=O)N(C)C)C2)=O)C1 39644,C1(C(=O)NCC2(OC)CCN(C(c3nnn(CC)c3C)=O)C2)CN2CCC1CC2 39645,C1(O)(CNC(C(C2CC2)OCC)=O)CN(C(c2csc(CC(F)(F)F)n2)=O)C1 39646,C(C1CN(C(=O)C2=CCCCC2)CC1C(=O)NCC(C)(C)CC)=CC 39647,N1(C(Cc2cccc(C)c2)=O)CCC2CCC12CNC(=O)C=Cc1cncs1 39648,C1(NC(c2ncc(Cl)cc2Cl)=O)COC2(CCN(C(C3(O)CCSCC3)=O)C2)C1 39649,CC1CCCc2ncc(C(N3CCCC(C)(NC(c4cc(=O)cc[nH]4)=O)C3)=O)n21 39650,CCCCCCC(C(=O)NCC1CN(C(c2scnc2Cl)=O)CC1O)NC(C)=O 39651,c1(C(=O)OCC)cc(=NCC(C2CC2)NC(C2CCCC3(CC3)C2)=O)[nH]c(C)n1 39652,C(=O)(C(C(=O)OCC)OC)NCC1(F)CN(C(C2(CC=C)CCC2)=O)C1.C(C)(C)(C)O 39653,N1(C(CCC=C(C)C)=O)CCc2ccccc2C1CNC(=O)CC1C=CCCC1 39654,C(=O)(C(CNC(C12CC(F)(C1)C2)=O)CC(C)C)Nc1c(COC)ncs1 39655,C1(NC(C2CCSCC2)=O)C2CCC(C2)C1C(=O)NC1CC2CC3C(C2)C13 39656,c1(OC)cc(C)ccc1CNC(=O)NCCC(C(=O)NC(C)(C)C)OC 39657,CCC(C)(CCC(C)C)C(=O)N(CC(C)(C)NC(c1n[nH]c2c1CC1CC21)=O)C 39658,Cc1cn2c(n1)CC(C(=O)NCC1(O)CCN(C(c3cscc3F)=O)CC1)CC2 39659,c1(C(=O)NC(CN(C(=O)CC(C)F)CC)C)c(C)c(O)nc2ccccc12 39660,C1(C)(C(=O)OC)CN(C(C2CCC2)=O)C1.C12(CC1)C(=O)N2 39661,C(=O)(C(=O)CCC(C)C)N1CCCCC(C(N2CC(C)C=C(C)C2)=O)C1 39662,c1(C(N2CCC(O)(C(=O)Nc3c(OC)nccn3)C2)=O)cccc2c1CCC2 39663,N1(C(=O)CCCC2CCOCC2)CCC2(CCCN2C(=O)CCOC2CC2)C1 39664,c1(CC(=O)NCC2(O)CCN(C(C3CSCCS3)=O)CC2)cccc([N+](=O)[O-])c1 39665,C1(C)(CNC(C=NOC)=O)CC(F)(F)CN1C(c1ccc(C)nn1)=O 39666,C1(C2(O)CN(C(=O)CCC(F)(F)F)C2)(CNC(c2ccn3c2CCCC3)=O)CC1 39667,c1(C(C(=O)NC2CCN(C(c3nncs3)=O)CC2F)O)ccc2ccccc2c1 39668,c1(C(N(C)CC2CC2CC(=O)NC2CCC(CO)CC2)=O)n[nH]cc1[N+](=O)[O-] 39669,c1(OC)nn(C)cc1C(=O)NC1CC(CNC(C2(C3CCCO3)CC2)=O)C1 39670,c1(NC(C(=O)NCC2C(NC(c3c(C)scn3)=O)CC2)=O)ccc(Cl)cc1 39671,C(=O)(C(C)(C)C(C)NC(=O)C(F)OC(F)(F)F)NC(CCC=C)(C)C 39672,c1(CC(N2CC(CNC(C=CSC)=O)CC(C)(C)C2)=O)nccc2ccccc12 39673,C1(N(C)C(C2CNC(=O)C2)=O)CCCN(C(c2ccnc(O)c2)=O)CC1 39674,C1(C(C)C)(C(N2CCCCC2)=O)CCN(CC=CC2CCCC2)C1 39675,Cc1cc(Cl)ncc1NC(C1CC2CC2N1C(c1snnc1C)=O)=O 39676,C#CC1COCCN1C(c1ccc(OCCCC#N)cc1)C(=O)NCCOC 39677,CCCCCCC(F)C(=O)NC1CC2CCC(C1)N2C(c1ccc(Cl)o1)=O 39678,NC(=O)CC(O)C(=O)NCC1CN(C(=O)CCCCCF)CCC1C(F)(F)F 39679,CN1CC2(CN(C(C3(N(C)C(c4c[nH]nc4C4CC4)=O)CC3)=O)C2)C1 39680,C1(C(=O)NC2C(NC(C(c3cccc(C)c3)F)=O)COCC2)CC2CCC1CC2 39681,C=Cn1nccc1C(=O)NC(CC1CCC1)C(=O)NC1(CC)CCOC1 39682,c1(OC)ccc(C(O)C(N2CCC(NC(c3nc(C(C)(F)F)cs3)=O)C2)=O)cc1 39683,C1(C(=O)NC2C(CNC(c3coc(-c4ccccn4)n3)=O)COC2)CCCCO1 39684,C1(C(=O)NCC(C(C)C)NC(C2CCN(C(N)=O)CC2)=O)C2CCN1CC2 39685,Cc1cccc(-n2nc(CCN(C)C)nc2-c2cnn3ccsc23)c1C 39686,C1(NC(C2(OC)CCCOC2)=O)CCCN(C(=O)C=Cc2ccn(C)c2)C1C 39687,c1(NC(=O)NCC2CN(CCC)C(=O)C2)nccc(=NC(C)Cc2ccco2)[nH]1 39688,C1(C(N2CC(O)(CCC)C2)=O)(NC(=O)C(C)NC(C)=O)CCCC1C 39689,CC1(C)CCCC(NC(=O)CSCCNC(=O)CC2CC=CCC2)C1 39690,C(=O)(C(COC)CC(C)C)NCCCN(CCC)C(C1CN2CCC1CC2)=O 39691,c1(CC(=O)NCC2(C(=O)NCc3ccc(O)nc3)CC2)ccc(O)cc1 39692,N1(C(C23OCC(C)(C2)C3)=O)CCC(C2CC2)(CNC(=O)CCCC2CCC2)C1 39693,N1(C(C2(CC#C)CCCO2)=O)C2CCC(C2)C1C(=O)NC1C(O)CC1O 39694,c1(C(=O)NC2CN(C(C=Cc3cn(C)nn3)=O)C2)cc(F)c(Br)c(Cl)c1 39695,Cc1cncc(CC(=O)N(C(C)CN(C(=O)CC2CCCC(=O)C2)C)C)c1 39696,C1(CC(=O)N(CC(CNC(C(COCC)C)=O)C)C)CCCCC1(C)C 39697,c1(C(=O)OCC)ccc(NC(C2CCN2Cc2coc(C)n2)=O)cc1F 39698,C12(C(=O)NC(C3(OC)CCCC3)(C)C)CC(C)(CN1C(=O)OC(C)(C)C)C2 39699,N1(C(c2c(C(=O)OC)nccc2)=O)CC2CC1CCN2C(C1(F)CCCCC1)=O 39700,C1(NC(C(C2CCN(C(c3ccc(CC)nc3)=O)C2)(C)C)=O)CNC(=O)C1(C)C 39701,C1(CNC(=O)OC(C)(C)C)CCN(C(=O)NC2(CC)CCOCC2)CC1OC 39702,C1(F)(CNC(c2scnc2Cl)=O)COCCN(C(C2OCCCO2)=O)C1 39703,CCCC(C)(O)CC(=O)N1CC(NC(c2cnc(C(C)C)s2)=O)C(CC2CC2)C1 39704,c1(OCC)ccc(C(=O)NCCCCCCN(C(=O)CN2CCC2C)C)cn1 39705,c1(CC(=O)NCC2CCCOC2)cn2cc(-c3ccncc3F)ccc2n1 39706,CC(O)C(F)(F)C(=O)NCCC(C)(C)CNC(=O)CCOCc1ccncc1 39707,N1(CCNC(c2cc(CNC(c3cnn(CCF)c3)=O)[nH]n2)=O)CCCOCC1 39708,C12(NC(c3c(CC)c[nH]c3)=O)CCN(C(C3(CC4CC4)CC3)=O)CC1C2 39709,C1(C(N(C(c2ccccc2)C(C)C)C)=O)CCC1(F)F 39710,N1(C(Cc2cc(C(C)C)no2)=O)CCC(NC(=O)C(F)C(C)(C)O)C(CO)CC1 39711,C=CCC(F)(F)C(=O)NC1CC2CC1CC2C(=O)NCCc1nc[nH]n1 39712,C(=O)(C(F)CC(C)(C)NC(C1CC(=O)CC12CCC2)=O)NCC(=O)NCCC 39713,C(=O)(C(F)CC(C)(C)NC(C1(C)CCCCC1C)=O)NC(c1ncccn1)CC 39714,c1(C(C)=O)c[nH]c(C)cc1=NC1CCc2ncc(C(F)(F)F)cc2C1 39715,c1(OC)ccc(CNC(=O)C(N)Cc2cc(Cl)ccc2Cl)c(F)c1F 39716,CCC(CC(=O)N1CC2CC1CN(C(=O)C(C)(C)S(C)(=O)=O)C2)C(C)(C)C 39717,O=C(CCCCC(F)F)NCCC1CSCCN1C(=O)C(O)CC1CCCCC1 39718,C1(COC(c2c(SCC)cccc2)=O)CCN(C(=O)CCc2ccc[nH]2)CC1F 39719,N1(C(c2cccc(CC)c2C)=O)CCC12CCN(C(c1cc(C(=O)O)c[nH]1)=O)CC2 39720,c1(CCC)cc(Cl)nc(NC(=O)C(N2CCCC(OC)C2C(=O)OCC)=O)n1 39721,C(CNC(=O)CC1(C)CCOC1)(CCNC(c1[nH]cnc1C)=O)OC 39722,C1(CNC(C=CCC)=O)CCC12CCN(C(=O)C=CS(F)(F)(F)(F)F)CC2 39723,N1(C2CCN(C(c3cc(COCC)[nH]n3)=O)C2)CCN(C(=O)CC(C)CF)CC1 39724,C(c1cncc(O)c1)=CC(=O)NCC1N(C)CCN1C(=O)CCC(N)=O 39725,N#CC1CC2(CC(NC(=O)CCC3CCCN(C(c4sccc4CO)=O)C3)C2)C1 39726,c1(C(N(C(C)C(=O)NC(C)Cc2ccncc2)C(C)C)=O)cc[nH]c1CC 39727,CCCC(O)(CCC)CC(=O)N1CCN(C(C2COC(C)C2)=O)C2(CCC2)C1 39728,CC1CCN(C(=O)CSCc2ccccn2)CC1CNC(=O)Cc1n[nH]c(=N)s1 39729,C1(NC(C(C)NC(=O)C2CC2)=O)C2CC3C(C2)C13C(=O)N(CCC[Si](C)(C)C)CO 39730,C1(CNC(=O)COCCF)CC2CN(C(c3cncc(-n4ccnn4)c3)=O)CC12 39731,N1(CC)CCC(N(C(c2ccn(CCOC)n2)C(=O)NC)C)C(C)C1 39732,CC(C(=O)NC(CNC(=O)C(=O)NCc1ncc[nH]1)CO)n1ccnc1 39733,N1(C(=O)C2=CCCC2)CC2=C(C1)CN(C(C1(c3ccc(F)cn3)CC1)=O)C2 39734,Cn1nc2c(c1C(N1CCC1CNC(=O)CC1(CO)CCCC1)=O)CS(=O)(=O)CC2 39735,C12CCCN(C1)C2=O.C(=O)(C(C)COC(C1CC(O)(C(F)F)C1)=O)N(CC)CC 39736,C1(N(C(=O)CSc2ccccc2)CC)CCCN(C(c2ncnn2C2CC2)=O)C1 39737,c1(C(C)C)ncc(C(=O)NCC(C)(F)CNC(=O)CNc2ccccn2)s1 39738,c1(OC)cnnc(C(=O)NC(C)CCCNC(=O)C(C)OCC2CC2)c1 39739,C(C1=CCN(C(c2ccccc2C)=O)CC1)NC(C(C1CCC(=O)NC1)CC)=O 39740,C(CCCCC(=O)N1CCC(C(=O)NCC2CC2(Cl)Cl)C1(C)C)OC 39741,Cc1ncc(C=CC(N2CC=CC(NC(C3(C)CCCOC3)=O)C2)=O)s1 39742,c1(C(C(=O)NC2CC(CCNC(c3cnc(CC)s3)=O)C2)(F)F)ccccc1F 39743,C1(CNC(CCNC(N)=O)=O)CCCCC1NC(C12CC(CF)(CO1)C2)=O 39744,Cc1[nH]c2ccccc2c1C(=O)NC(C)C(C)NC(c1cc(F)c(N)cc1F)=O 39745,C1(C(=O)NCCC2CNC(=O)O2)CC1C1CCN(C(=O)C2=CCCOC2)CC1 39746,N1(CC(n2cc(-c3ccc(F)nc3)nn2)C)CCC(C#N)(C(=O)OC(C)(C)C)C1 39747,C1(CNC(CCC(=O)OC)=O)COC(C)(C)CN1C(C1CC2CCC(C1)N2C)=O 39748,N1(C(c2nnn(C)c2C(F)F)=O)CCC2CCN(C(c3cccc(Cl)c3)=O)CC12 39749,c1(C(=O)NCC2(CCCNC(C(C(C)C)O)=O)CCCC2)nc(O)nc(O)c1N 39750,N1(C(C(CC)=CC)=O)CCC2(CCCCN(C(C34CCC(F)(CC3)C4)=O)C2)C1 39751,N1(C(C2(CCC)CC2)=O)CC(C)(C)C(NC(=O)CC(C)(C)COC)C(C)(C)C1 39752,C12(CNC(c3nc(Cl)cs3)=O)CN(C(=O)CCc3ccccn3)CC1(C(F)(F)F)C2 39753,C1(CCC)CN(C(=O)CC2CCSC2)CC1C(N1CCC(C(=O)OCC)C1)=O 39754,c1(OC)cnccc1C(=O)NCCC1CCCCN1C(c1cc(C(C)=O)c[nH]1)=O 39755,c1(C(N2CC(NC(CCCC3CCC(C)C3(C)C)=O)C2)=O)c2ccccc2nn1C 39756,C#Cc1cc(F)c(C(N2CC3CC3(NC(C3COC3)=O)C2)=O)cc1F 39757,O=C1COc2cc(C(N3C4CCC3CN(C(C3CCC5CC35)=O)C4)=O)ncc2N1 39758,N1(C(CCC2CCC(NC(C(C=C)(C)O)=O)C2)=O)CCC2(CCC2)C(O)C1 39759,C1(C(=O)NCC23CC(NC(c4ccn(C)n4)=O)(C2)C3)CCC(F)CC1 39760,c1(C(=O)NCC(CCC)C(=O)N(CCC(F)(F)F)C)ncn2ccccc12 39761,CC(C)CCCC(C)C(=O)Nc1nc(=N)nc(N2CCC(N3CCC(O)C3)C2)[nH]1 39762,C1(CNC(c2c(C)occ2C(F)(F)F)=O)CC(F)(F)CN1C(c1c[nH]c(=N)s1)=O 39763,c1(CC)nc(C(=O)NCC2(NC(=O)Cc3ccnc(C(N)=O)c3)CCC2)c(C)o1 39764,c1(C(=O)NCC(CC)NC(=O)CCCOC2CCOCC2)occc1C(C)C 39765,C1(C)(NC(c2c(OC)c[nH]n2)=O)CCN(C(c2cccc(I)c2)=O)C1 39766,C1(C(N2C(CCNC(Cc3c(C)cnn3C)=O)CSCC2)=O)Cc2cscc2C1 39767,C1(N(CC(C)C)C(=O)COC2CCCC2)CCN(C(C2CC(F)C2)=O)C1 39768,C(c1cc(C)ccc1OC)=CC(=O)N(CCCCNC(CC(COC)C)=O)C 39769,N1(C(COCC(=O)NC)=O)CCCCC(C(=O)NCCCCC(C)(C)C)C1 39770,Cc1ccc(C(N2CCCC2C(C)(C)CNC(C2OCC2(C)C)=O)=O)nc1 39771,c1(CCCC#C)ccccc1.c1(N)ccccc1 39772,c1(C(N(C(C)CCNC(C2CC(N(C)C)C2)=O)C)=O)ccn(C(C)(C)C)c1 39773,c1(NC(c2cc(C)sc2)=O)cnn(C)c1C(N1CCN(C(C)C)CC1)=O 39774,C(C)(CCCCNC(=O)CCc1nnc(C2CCCC2)o1)NC(C1C(C)C1C)=O 39775,Brc1c(NCC2CCCCC23CCC3)nc2ccc(C3CC3)cn12 39776,N1(c2cc(C)nc(C3CCC3)n2)CCC(C)C(NC(=O)CC2CC=CCC2)C1C 39777,C1(O)(CNC(C)=O)CCCN(C(=O)CC(O)C(C)C)C1 39778,c1(C(=O)OC)cncc(OCCNC(C2(C)CC2F)=O)c1 39779,CCCCCS(=O)(=O)CC(=O)NCC1(OC)CN(C(=O)C(C2CC2)N(C)C)C1 39780,c1(CCC)c(NC(N2CCCC(CF)C2)=O)nnn1Cc1ccccc1Cl 39781,c1(C(=O)NC2(C)CCN(C(c3cn4ccsc4n3)=O)C2)ccc(Cl)nc1O 39782,c1(CCNC(C2N(C(CS(C)(=O)=O)=O)CCC(O)C2)=O)ccc(S(=O)(=O)F)cc1 39783,C(=O)(C(CC(C)C)NC(C)=O)NC1C2CCN(C(C3(CC)CCNC3=O)=O)C21 39784,N1(C(c2ccn(CCCC)n2)=O)CCC(C)C(CNC(=O)C#CC(C)(C)O)C1 39785,N1(C2CCN(CCCN=[N+]=[N-])CC2)CCN(C(C2NC3COCC23)=O)CC1=O 39786,c1(N(C)Cc2ccoc2)ccc(S(=O)(=O)N2CCn3ncc(CO)c3C2)c(Br)c1 39787,c1(C(N)=O)ccc2c(c1)OCCN(C(c1cc(Br)c(F)cn1)C(=O)NC1CC1)C2 39788,n1(C(C(=O)N(CCNC(=O)CN(CC(C)(C)C)C)CC)C)ccc(C)n1 39789,c1(OC)ccccc1N(C(c1cccnc1OC)C(=O)NCc1cccs1)C 39790,C(=O)(C1=C(C#N)CCC1)NCC1CC(C)(C)CN1C(=O)COC(F)F 39791,C1(C(N2CCC(n3cc(C(N4CCCC4)C)nn3)C2)=O)CCc2nncn2CC1 39792,Cc1ccncc1CCNC(=O)CC1CC(NC(C2C(C#N)C2(C)C)=O)C1 39793,C1(C(=O)NCC(C=C)O)CC12CC(NC(c1c[nH]nc1C(F)F)=O)C2 39794,CC(C)CC(C(=O)NC1CC2C1CCN2C(=O)CC1CN2CCC1CC2)C(N)=O 39795,c1(OC)cccc(NC(=O)NCC2(NCc3cc(Cl)ccn3)CC2)c1 39796,C1(CNC(CSc2n(C)ccn2)=O)CCCCN1C(c1cn(C2CC2)cn1)=O 39797,N1(C(C2NC(=O)OCC2)=O)C2CCC1(CNC(c1cnn(CCO)c1)=O)CC2 39798,c1(C(C2(CC#N)CC2)NCC(CC)C)nnnn1CC(F)F 39799,N1(C(=O)NC(c2cccc(Cl)c2)CC)CCC2(CSC2)C1 39800,Cc1ccc(F)c(O)c1C(=O)NC1CCCCN(C(=O)CCc2cscn2)C1 39801,N1(C(CCCCOC)=O)CCC(C)(C)C(NC(=O)C(C(C)CC)NS(C)(=O)=O)C1 39802,C1(N(C(CC(C)=C(C)C)=O)C)CCCC(N(C)C(c2c[nH]nc2Cl)=O)C1 39803,C1(CNC(C2(C)CC2C(F)(F)F)=O)CCCN1C(=O)CC1CCOC1=O 39804,Cc1cc(C(C)NCC(C)CCCO)ccc1[N+](=O)[O-] 39805,c1(OCC(=O)NC(C(C)NC(=O)CC2CCCCC2)CO)cccc(F)c1 39806,C1(CC(N2CCC(CN(C(=O)CCC3CC3)C)C2)=O)CCCCCC1 39807,C1(CC(N2CC(CC=C)(NC(CCCC#C)=O)C2)=O)NC(=O)CN(C)C1=O 39808,C1(CC(=O)NC2(CNC(CN(C(CCOC)=O)C)=O)CC2)CC2CCC1O2 39809,C(CCC(=O)NC(C(=O)NC12CCCC1C2)c1cccs1)=CC(C)C 39810,C(=O)(C(C)(C)CCC#N)NCCC(C)N(C)C(C1OCCN(C)C1=O)=O 39811,C(C)(CCCC(=O)N1CCOCC1C1CC1)NC(COCCCC(C)C)=O 39812,Cc1cc(CNC2CC(C(=O)NCCN3CCS(=O)(=O)CC3)C2)c(O)c(Br)c1 39813,c1(C(=O)NC2CN(C(C(CO)NC(N)=O)=O)C2)cc(Cl)c(Cl)cc1N 39814,C=CCCCCCC(=O)NC(C(=O)NC1CC(C)(C)OC1(C)C)C1CC1 39815,Cc1ccc2n[nH]cc2c1C(N1CCN(C(c2cccn2C(C)C)=O)C(C)C1)=O 39816,N1(C(C2CCC2)=O)CCCC2C1CCN2C(c1sccc1F)=O 39817,N1(C(C(CC=C)NC(C)=O)=O)CCC(C(=O)NCc2nccs2)C1(C)C 39818,C1(F)(C(=O)NC2CN(C(C3C(C(C)C)CCC3)=O)C2)C(C)(C)C1(C)C 39819,CC1CCCC(OCC(=O)NC2CC(c3ccccc3)(NC(=O)COCF)C2)C1 39820,c1(C(=O)NS(CCC(C)(C)C)(=O)=O)cc2cc(F)ccc2cn1 39821,C12(COC)CN(C(=O)C3=CCC3)C(CNC(c3ccc(C)s3)=O)(C1)C2 39822,CC1OC(C)C(C(=O)NC(C2CCN(C(C3CCCS(=O)(=O)C3)=O)CC2)C)C1C 39823,Cc1cc(N(C2CCN(C(C3(O)CCOCC3)=O)C2)C)c(C#N)cn1 39824,C(=O)(C(F)CC(C)(C)C)N1C(CC(=O)NC(C(=O)OC)C2CCC2)CCC1 39825,c1(C(N2C(C(C)(C)NC(CCc3onc(C)n3)=O)CCC2)=O)cc(Cl)nn1C 39826,C(=O)(C1=NOC(C)C1)N(C(C)C(=O)NCC1(C)CC2(CC2)C1)C1CC1 39827,c1(OC)c(C(=O)NC2COC(C(F)F)C2)ccc([N+](=O)[O-])c1F 39828,N1(C(c2c(OC)nsc2)=O)CCC(C=CC(=O)NCCC(O)C(F)(F)F)CC1 39829,Cc1cc(C2CC2)ncc1C(=O)NC(C1CN(C(c2ccncc2Cl)=O)C1)C 39830,Cc1cnc2ccc(C(=O)N(C)Cc3cccnn3)cn12 39831,O=C(NN1CCCC1C(=O)N(C1CC1)Cc1nc[nH]n1)C1CC(CCCF)C1 39832,N1(C(CNC(C2C(C)C2)=O)=O)CCCCC1C(=O)NCC12CCN(CC1)C2 39833,c1(C(=O)OCC)cc(CNC2CCN(C3CCNCC3)CC2)nn1C 39834,C#CC(Cn1cccn1)NC(=O)CC1CC(N)C1 39835,c1(C(C)C)cc(C(F)(F)F)nc(NC2(CNC(=O)C(F)=CC3CC3)CC2)n1 39836,C1(C(=O)NCCCNC(C(C)c2ccon2)=O)CSc2ccccc2O1 39837,N1(C(c2ccc(CCC)[nH]2)=O)CC(NC(c2cc(O)nn2C)=O)C(C)C1 39838,C(=O)(C(F)(F)C(F)F)NCC(C)CNC(=O)CC1(N(C)C)CC1 39839,C(=O)(C(F)CC(C)(C)NC(c1ccc(F)cc1C)=O)NC(C#C)CC(C)C 39840,CN1CCN(C(=O)C(C2(O)CCCC2)F)C(CNC(=O)CCC2CCC2)C1 39841,C1(C(=O)NCC(CC)NC(c2ccc(CO)cc2)=O)CCCCC1C(F)(F)F 39842,C1CCC(=O)NCC2CC(CO2)CNC1=O.C1(C)(SC)CCCC1 39843,c1(CC)cc(-c2nc(C)nn2CCOc2cccc(C)c2C)ccc1O 39844,c1(OC)cc(C=CC(=O)NC2CC(NC(=O)C(O)C3CCC3)C2)ccc1O 39845,C=C=CCCC(=O)NCC(=O)NC1CCCC1.c12noc-1n2 39846,c1(CC)[nH]nc(C(=O)NC2(C(=O)NCCCN(C)OC)CCCC2C)c1C 39847,N1(CC(=O)NCC2CCC3(CCC3)O2)CCC2(C=CCO2)CC1 39848,c1(CC(=O)OC(c2ccccc2)C)c(F)cccc1F 39849,c1(C(C(=O)NC(CCCNC(Cc2c(C)n[nH]c2C)=O)C)O)ccc(Cl)cc1Cl 39850,n1(CC(=O)NC2(C3CN(C(C4(C)CC=CCC4)=O)C3)CC2)ncc2ccccc12 39851,C1(C(=O)NC2CON(CC)C2=O)CN(C(C2CC3(CC3)CO2)=O)CC1(C)C 39852,N1(C(c2cc(C)n(C(C)C)n2)=O)CC(CNC(c2n[nH]cc2Br)=O)OC(C)(C)C1 39853,NS(=O)(=O)C1(C(=O)NCC2CC3CCC2N3C(=O)C2=CCCO2)CCCC1 39854,c1(NC(CC2OCC(C)OC2)=O)cc2oc(=O)[nH]c2cc1F 39855,Cc1cccc(C(=O)NCC2CCCC2NC(c2c(F)cccc2F)=O)c1C 39856,c1(C(=O)NCC2N(C(c3ccn(CCCC)n3)=O)CC=C2)cnc(S)n1C 39857,C(=O)(C(C)(C)CS(C)(=O)=O)NCCC1N(C(C(COC)COC)=O)CCCC1 39858,n1(CCOCCNC(C(c2cccnc2)C)=O)cc(C2CC23CC3)nn1 39859,Cc1ccn2c(C(=O)N(CC(C)(C)CNC(=O)CC(=O)NC3CC3)C)cnc2c1 39860,c1(C(=O)NCC2CN(C(CNC(c3cn(CC)nc3)=O)=O)C2)cccc(Cl)c1Cl 39861,c1(C(N2CCC(NCc3ccc(OC)c(OC)c3)C2)=O)cc2c(s1)CCOC2 39862,C1(C(=O)NCCc2cn(CC)nn2)C=CCCN1C(=O)CCCCOC 39863,C1(NC(C2(C#C)CCCC2)=O)CC2CC1N(C(=O)C(CC)=CC)C2 39864,C(CN=C(NCCc1ccc(F)cc1F)NCC1CCCCO1)c1ccc(C)o1 39865,C1(c2n(C)cnc2)CN(C(=O)CSS(C)(=O)=O)CC1CNC(=O)C=CBr 39866,Cc1nc(O)ccc1C(=O)NCCc1cc(C(=O)N(C2CCC2C)C)no1 39867,Cc1cc(NC23CCCC2CN(C(=O)CO)C3)n2ncnc2n1 39868,N1(C(C23N(C(C(C=C)C)=O)CCC2C3)=O)CC2(CC(CO)CO2)C1 39869,N#Cc1ccc(-c2cn(C3CCCN(C(c4sccc4CO)=O)C3)nn2)s1 39870,C1(C(=O)NCC2(CCNC(C3(N(C)C)CCCCC3)=O)CC2)CCCCC(=O)C1 39871,c1(C(N(C(CNC(C2C(C)C2)=O)C)C)=O)ccc(N2CCC(C)CC2)nc1 39872,c1(C(=O)NCC2(F)CC(NC(C3(COC)CCOC3)=O)C2)ccncc1OC 39873,Cc1cccc(C)c1CCNC1(c2nnnn2CCC2CC2)CC(NC(N)=O)C1 39874,C(N=c1nc(C(=O)NC)cc(C)[nH]1)c1ccc(CNC(CCOCC)=O)c(F)c1 39875,N1(C(C(N(C)C)C2CC2)=O)CC(NC(c2cc(Cl)c(F)cc2F)=O)C(N=[N+]=[N-])C1 39876,N1(C(CCCOC)=O)CCCC(CO)(CNC(c2ccon2)=O)C1 39877,c1(C(=O)NCC2(NC(C3CCN(C)CC3)=O)CCOCC2)cc(F)ccc1N 39878,N1(C(=O)CCC2CCC2)CCC(n2cc(CCN3CCCC(Br)C3)nn2)CC1 39879,C(=O)(CCC(C)(C)O)NC(C1CN(C(=O)C2=CCCCC2)C1)C 39880,c1(COC)ccc(F)cc1C(=O)NCC1(C(C)NC(=O)CSC2CC2)CC1 39881,N1(C(c2cncc(N)c2)=O)CCN(C(c2cc3c[nH]nc3s2)=O)C2CC12 39882,C(=O)(C(=O)CC(C)CC)N(C(C)C(=O)NCC1CCCCCCC1)CCC 39883,c1(C(=O)NC2CCC(NC(c3c(CC)nns3)=O)CC2)cc2c[nH]cnc-2n1 39884,n1(CC)c(=O)c(C)nc2cc(C(N3CC(NC(C4CCC4CF)=O)C3)=O)ccc12 39885,Cc1cc(CCCC(=O)N(CC(C)NC(=O)C=Cc2ccccn2)C)c(C)s1 39886,CC1(C)CCC2(CN(c3ccnc(N4CC5C(C4)C5(F)F)n3)CCO2)C1 39887,C(=O)(C1=NNC(=O)CC1)N1C(CNC(c2c(Cl)nc(OC)s2)=O)C(C)CC1 39888,S(=O)(=O)(c1[nH]c(=NC(C)Cc2ccccn2)ccc1Br)NC(CC)(C)C1CC1 39889,c1(-c2cnc(NC(C(C)(C)Br)=O)s2)cccc2cc[nH]c12 39890,CCC(C)(C#N)C(=O)NCC1CCN(C(=O)CCc2nnc(C3CC3)o2)CC1 39891,C(=O)(C(C(C)C)NC(=O)OC)NCCN(C(CCC=CC)=O)CC 39892,c1(SC)c(C(=O)NC2CCCCC2NC(c2cnn(CCO)c2N)=O)cnn1C 39893,C1(C2CCOCC2)(C(N(C)CCN2CCN(C(=O)CNC(N)=O)CC2)=O)CC1 39894,C1(C(=O)Nc2cccc(NC(C3(C)ON=C(C)C3)=O)c2)CCc2nnnn2C1 39895,C1(CC(=O)N(CCOCCN(C(C(C)N(C)C)=O)C)C)CCCSC1 39896,C(=O)(CC(C(=C)C)OCC)N1CC(C2CN(C(CC3CC(=C)C3)=O)C2)OCC1 39897,c1(C(=O)NC2CCN(C(C(CC)OCC)=O)C2)cc2n(n1)CCO2 39898,C1(NC(C2N(C(C)=O)CCC2)=O)CC2(C1)CN(C(=O)CC1C(=O)N(C)N=C1C)C2 39899,C(=O)(C(F)C(=O)NC1CC(CNC(=O)Cc2cc(=O)n(CC(C)C)[nH]2)C1)OCC 39900,Cc1ccc(CNC(C2(c3cc[nH]n3)CC2)=O)cn1.C12(CCC1)C(=O)NC2 39901,N1(C(c2ccnc(OC)n2)=O)CCC2(CNC(=O)C(C)=C3CCC3)CCCCC12 39902,C1(C(N(CCNC(C2CCCC(C)(C)C2)=O)CC)=O)CC12CCCCCC2 39903,C(=O)(CCCCC(F)(F)F)N1CC2C(NC(c3ccc(N)c(F)c3F)=O)C(C2)C1 39904,n1(CC)cc(Br)cc1C(=O)NCC1CC1NC(C1(NC(N)=O)CC1)=O 39905,C1(CC=C)CCCCC1C(c1ncnn1C(C)C)NCc1nnnn1C1COC1 39906,C=C=CCCOC(C)(C)C.C1(=O)C(C)ONC(=O)OCCN1 39907,Cc1cc(CNc2ncc(C(=O)OC(C)(C)C)cn2)c(O)c(Br)c1 39908,c1(C(=O)NCCOCC(=C)C)cccnc1CNC(=O)CN1CCCCCC1 39909,c12ccc3nc([nH]c3c1)OCC(=O)N2.C1(CCCC)CCCC1C(=O)OC 39910,C1(NC(Cc2c(C)scc2)=O)CCCC(NC(=O)C(C)(C)Br)C1 39911,c1(C(=O)NC2CC(C)(NC(=O)CCC3CCOC3)C2)cc(N)c(F)cn1 39912,C(=O)(CC(F)(F)F)N(CC(C(=O)NCC(=O)OC(C)C)C)C 39913,CC1=C(C(=O)NCC2CCCN2C(C2(C(F)(F)F)CCC2)=O)CCO1 39914,C1(C(=O)NCCn2c(C)ncc2)CCCN(C(C2C=CCC2)=O)CC1 39915,N1(C(CC(=O)OC)=O)CCOC2CN(C(c3n[nH]c4cc(C)ccc34)=O)CC12 39916,C1(NC(c2n[nH]c(C)c2O)=O)CN(C(=O)CC(C)(C)c2ccccc2)CCC1C 39917,N1(C(=O)Nc2ccc(Cn3cccn3)c(Cl)c2)CCc2[nH]ccc2C1 39918,C(=O)(C(CC1CC1)NC(=O)CC=CC(C)(C)C)N1CC(CCC#C)C1 39919,c1(OC)ncc(C(N2CC(NC(=O)CN(C)C3CC3)C(O)C2)=O)cc1F 39920,c1(N(C)C(c2cscc2-c2cc(O)cc(C#N)c2)=O)nc2ccccc2s1 39921,N1(C(c2c(C)nc(C)[nH]2)=O)CCN2CCOCC2(CNC(=O)CC(C)F)C1 39922,c1(C(=O)NCC(CC)(CC)NC(=O)C(F)CC(C)C)snc2ccccc12 39923,C1(CC)CN(C(C2CCCC(C#N)C2)=O)CCN1C(=O)CCCc1ccccc1 39924,c1(C(=O)NC2C(NC(CC(COC)C)=O)C2)cccc(=O)n1C 39925,Cn1cnc2nc(=NCC3CCCC(NC(=O)COC(F)F)C3)[nH]cc12 39926,N1(C(C2(C)C=CCN2C(=O)CN2CCSCC2)=O)CC2CC1CC2CF 39927,N1(c2cc(C)ncn2)CCCC12CCN(C(c1cccc3c1ncn3C)=O)C2 39928,C1(C(N2CC(c3n(C)ccn3)C(NC(=O)C3=CCC3)C2)=O)Cc2cscc2C1 39929,N1(C(c2occ(C)c2)=O)Cc2ccccc2C(NC(c2ccc(N)c(O)c2)=O)C1 39930,C(c1ccccc1F)=CC(=O)NC(C)CC(C)NC(=O)C1=C(Cl)CC1 39931,C1(NC(CCC=CC(C)C)=O)CCN(C(c2cn(CC(F)(F)F)nn2)=O)C12CC2 39932,CC1CCC(=CC(=O)NC(C)CNC(=O)C(C)N2CC(C)C2)CC1 39933,C1(C(N2CCOC(CCNC(c3cccc(Cl)c3)=O)C2)=O)(CSC)CCOCC1 39934,N1(C(c2nc(C(C)(C)C)sc2)=O)CC2(C1)CN(C(=O)CC1(C)CC1(Cl)Cl)C2 39935,C1(C(N(CCCCN(C)C(C2(CO)CC(C)(C)C2)=O)C)=O)CCC2(CCC2)OC1 39936,CCC(C)C(O)C(C)C(=O)NCC1(NC(=O)Cn2cc(C(=O)NC)nn2)CCC1 39937,C1(NC(c2ncn(C(C)C)c2)=O)CN(C(C2(O)CCOC2)=O)CC1C 39938,N1(C(c2c(C)cno2)=O)CC(NC(c2c(C)ncn2O)=O)CC12CCCCC2 39939,CC(C)(C(=O)NC1CN(C(=O)CC(=O)NC2CC2)C1)C1CCCO1 39940,c1(OC)c(C(=O)NC2CN(C(c3c(N)cccc3Cl)=O)C2)oc2ccccc12 39941,C1(CC)C(C(=O)NCc2ccc(C)cc2)CCN1C(=O)C(C)O 39942,N1(C(CCC(=O)NC)=O)CCC(C2CC2)C1CNC(c1cnc(C)c(OC)c1)=O 39943,c1(OC)ccc(C#N)cc1NCc1nc(Nc2ccc(F)cc2)[nH]c(=N)n1 39944,N1(C(c2cccc(CNC(CCCCC#C)=O)n2)=O)CCC2C(CCN2C)C1 39945,c1(C(N(CCN(C(c2cncc(NC)c2)=O)C(C)C)C)=O)nc[nH]c2ncnc1-2 39946,c1(C(C)(C)NC(c2ccncc2)CF)ccnc(Cl)c1F 39947,C(=O)(C1CCc2cccc(F)c21)N1CC(COC)OC(C)C1 39948,C(CC1=CCOCC1)NC(C(CC)N(C)C(c1cn(C)c(=O)cn1)=O)=O 39949,C1(NC(=O)CCc2cnc[nH]2)CCC12CCN(C(c1cc(Cl)ccc1O)=O)CC2 39950,N1(C(Cc2nc(C)sc2C)=O)CCCN(C(=O)CC(C)c2ccco2)C(CO)C1 39951,N(C(=NCCC)NC1CC(CC(N)=O)C1)C(C#C)CC 39952,C1(NC(N(CC(C(C)C)(F)F)C2CC2)=O)CCC2(CCOCC2)C1 39953,Cc1ccc(CC(=O)NCC(C(C)(C)C)NC(=O)CC2(O)CCOCC2)c(C)c1 39954,N1(C(CCc2scc(C)c2)=O)CC(C)CN(C(=O)CN2CCCCC2)C(C)C1 39955,C(C)(C)(CC(=O)NC(c1cn(C)nn1)C)NC(C=CCCC)=O 39956,c1(C(=O)NCC2(C)CCC(NC(=O)CC(F)(F)F)C2)cc2cc(Cl)ccc2o1 39957,C(=O)(CC(C)C(C)(C)NC(c1cnc(N(C)C)o1)=O)N1CCC(C)(CCC)C1 39958,c1(CC(=O)NC(CCNC(C2(OC)CC2)=O)C)csc2ccccc12 39959,c1(C(=O)NC(C2CCN(C(c3csc(C)c3N)=O)CC2)C)ccn2nnnc2c1 39960,c1(C(=O)NC2CCN(C(C(C)N(C3CCCCC3)C)=O)C2)cn2cnnc2cn1 39961,C1(NC(c2ccn(CC(C)C)n2)=O)CCN(C(=O)CC2CCC2)C1C1CC1 39962,CCC(C(=O)NC(CNC(=O)CC(C)N(C)C)CC(F)(F)F)C(C)(C)CC 39963,C(=O)(CCC(C)(F)F)NCCN(CCC)C(c1c(Cl)cncc1Br)=O 39964,CC1Cc2ccccc2N1C(=O)CC1(NC(C2C(C(=O)O)C2(C)C)=O)CCC1 39965,CC(C)(CC(=O)NC1CCC(CNC(C2CCCC3CCCN23)=O)C1)C(F)F 39966,C1(C#N)(C(=O)NCC2CCC(NC(c3scc(C)c3Cl)=O)CC2)CC12CCCC2 39967,C1(C(=O)NCc2cn(CC)nn2)CCC(C)(C)N(C(C2CCCCN2C)=O)C1 39968,c1(CC(=O)N(C)CC2CCCN2C(C23CC(F)C2C3)=O)cc(Cl)sc1Cl 39969,CC(Cl)(Cl)C(=O)N1CCC(C(C)(C)NC(C2CCC(C(=O)OC)O2)=O)C1 39970,N1(C(c2cnc(C3(CC)OCCO3)s2)=O)CCN(C(=O)C(C)(C)O)CC1C1CC1 39971,C1(OC)(CNC(C2C3CCCOC23)=O)CCN(C(=O)Cn2ncccc2=O)C1 39972,C#CCCC(C(=O)NCC(c1ccco1)O)NC(=O)C=C1CCC(C)CC1 39973,C1(C(=O)NC(CC)COC)CC(=O)CN1C(c1cccn1CC)=O 39974,c1(OC)ccc(C#N)cc1NC(=O)C(F)C1CC(C(=O)OC(C)(C)C)C1 39975,C(=O)(C(F)C(F)(F)F)NCC1(F)CN(C(C(C)CO)=O)C1 39976,C1(C(=O)NC2(CNC(c3ccc(C#N)cn3)=O)CCOC2)C2(CCC2)C12CCC2 39977,N1(C(C(C(COC)C)C)=O)CCCC2(NC(C3CCCCC3C)=O)CCCC12 39978,O=C(C1=C(Cl)CCOC1)NC1CC(NC(c2cc(C(F)(F)F)nn2C2CC2)=O)C1 39979,c1(CC)ccccc1C(N1CCC(CCC(=O)NC2CCOCC2OC)C1)=O 39980,N1(C(C(C)NS(C)(=O)=O)=O)CCC(F)(CNC(=O)CNC(C2CCC2)=O)C1 39981,N1(C(C2=CCCCC2C)=O)CC2(C1)CN(C(C1(CCN(C)C)CCC1)=O)CCO2 39982,C(=O)(C1=NOC(C)(C)C1)N1CC(NC(c2cnc(C(C)C)s2)=O)C(C)CC1 39983,C12(CNC(C(N3CCOCC3)C)=O)CCCCC1CN(C(=O)C(C)(C)CO)C2 39984,C(=O)(C(C)S(N)(=O)=O)N1C(CNC(C(C)C2CCC2)=O)CC(F)C1 39985,C1(C#CC(=O)NCC2CN(C(C3C4CC5C(C4)C35)=O)CC2(C)C)(CC)CC1 39986,C(CC)(C(=O)NC1CCC1C(=O)N(C(C)CC1CC1)C)=CCCC 39987,O=C(CC1=CCCCC1)N1CCC2(CC2C(N2CCCC2CCO)=O)C1 39988,Cc1ccc(C(F)C(=O)NCC(O)CNC(=O)CC2CCCCC2)cc1 39989,N1(C(c2ccc(C)s2)=O)CC2CCCCC2(NC(c2occ(C)c2C)=O)C1 39990,C1(O)(CNC(c2cc(-c3ccco3)no2)=O)CCCN(C(C2SCCS2)=O)CC1 39991,C1(=O)C(F)(C(C)C)CN1CC(C)(C)C.C1(C(C(=O)OC)=O)CCCCC1 39992,N1(C(C2CC(C)OC2)=O)CC2CN(C(c3ccc4nccn4c3)=O)CC(C1)O2 39993,N1(C(Cc2nc(COC)sc2)=O)CC2CC1CN2C(c1sccc1F)=O 39994,C1(C(=O)Nc2cn(CC)nc2)CC12CCN(C(=O)COC(C)=O)CC2 39995,C1(CNC(C2(C)ON=C(C)C2)=O)Cc2ccccc2CN1C(=O)Cc1ccns1 39996,N1(C(C(C)(C)c2ccccn2)=O)CC2CN(C(=O)CC3CCCCC3(F)F)C2C1 39997,Cc1ccnc(O)c1C(N1CCC(C)(NC(C2CN(C3CCOC3)C2)=O)C1)=O 39998,c1(OCC)ccc(C(=O)NCCCC2CCN(C(=O)CN(C)CCO)CC2)cc1 39999,CC1CCCN(C(C)CNC(=O)NC2CN(Cc3ncccc3C(F)(F)F)C2)C1 40000,C12(C(N3CC(Cc4cn(Cc5cn(C)nc5)nn4)C3)=O)CC3CC(CC(C3)O1)C2 40001,c1(C(N(CC(C)NC(CCN(CCC)C)=O)C)=O)noc2c1CCCCC2 40002,C1(C)(C(N2CC(O)(CN(C(=O)CNC(c3ccccn3)=O)C)C2)=O)C=CCCC1 40003,C(=O)(CCCN(C)C(=O)OC)NC(CNC(C1(C#C)CC1)=O)(C)C 40004,c1(CCC(N2CC(NCc3cc(Br)c[nH]3)C3(CC3)C2)=O)c[nH]c2ccccc12 40005,C1(NC(CCC(C)C)=O)CCCC12CN(C(C1(C)CCN(C)C1=O)=O)C2 40006,C1(C)(CNC(c2c(C)cno2)=O)CCCN1C(=O)CCSCC(N)=O 40007,Cc1noc(C)c1COc1ccc(C(=O)NCCC2CCN2C2CCCC2)cc1 40008,Cc1ccc(C(F)(F)F)c2c1N(C(N1CCCS(=O)(=O)CC1)=O)CCC2 40009,C(C)(CN=c1nc(C2CC2)[nH]s1)NC(COc1ccc(C)cc1)=O.C1C(=O)N1 40010,C1(C(=O)NC2(C(N3CC(N4CCCC4)C3)=O)CCN(C)C2)CCC2(CCC2)O1 40011,C1(n2cc(C(C)(C)O)nn2)CC2CCC(C1)N2C(c1cc(F)cc(Br)c1F)=O 40012,N1(C(c2scc(COC)c2)=O)CC(CNC(=O)CCC(F)F)CC1C 40013,C(C(O)C(=O)N1CC(O)(C2CCCN2C(=O)CCc2nc(=N)[nH][nH]2)C1)SC 40014,N(C1CCCc2c(F)cc(F)cc21)C(=O)CC1CCCO1 40015,N1(C(c2cnn(CC)n2)=O)CC(CO)C2(C1)CN(C(=O)CC(C)(C)CC(C)=O)C2 40016,N1(C(C2(CC=C)CN(C(c3cc(C)c(C)[nH]3)=O)C2)=O)CC(N(C)C)C(C)(C)C1 40017,N1(C(CC(CC)C(C)C)=O)CCC2CCN(C(=O)CCc3cc[nH]n3)C2C1 40018,N1(C(CC(=C)Br)=O)CCC2(CCCN(C(=O)CCOC3CCCC3)C2)CC1 40019,C1(CNC(c2n(C(C)C)cnc2)=O)CC(NC(=O)C(C2CCC2)N(C)C)CCO1 40020,Cc1c(C(=O)NC2CC2CNC(=O)CC2COCCO2)cc(Br)cc1N 40021,S(=O)(=O)(c1cccs1)NCCC(=O)NCC1(O)CN(C(C2(C)CC3(CC3)C2)=O)C1 40022,c1(C(C)NC(C2(CF)CCC2)=O)ccc(CNCc2nocc2C(C)(C)C)cc1 40023,Cc1ccc(C(=O)NCC2(NC(c3ccn(C4CC4)c3C)=O)CC2)nc1O 40024,c1(-c2cc(C(=O)OC3CC(C)(C)C3)n[nH]2)ccc(F)cc1 40025,N1(C(C2CCN(C(C)=O)CC2)=O)CC2CCN(C(=O)Cc3cnccn3)C2C1.C(C=O)N 40026,N1(CCONC(=O)NC2C=CCCCC2)C(=O)c2ccccc2C1=O 40027,N1(C(C2=C(C)CC2)=O)CC2CC(NC(c3nccc4n[nH]cc34)=O)C(C2)C1 40028,c1(C(=O)NC2C(CNC(C(CCC)OCC)=O)C2)cc(OCC)ccc1C 40029,C1(P(C)(C)=O)(C(=O)NCC2(NC(C(C)SCCCC)=O)CCCC2)CC1 40030,c1(OCCCC)ccc(C(=O)NC2CCCC2NC(c2n[nH]cc2Cl)=O)c(O)c1 40031,C1(C(N2CC(CC)(CC)C2)=O)CCN(C(c2cnn(C3CC3)c2)=O)C(C)(C)C1 40032,c1(C(=O)OC)sc(C(N2CCC(NC(C3(CC(F)F)CCC3)=O)CC2)=O)cc1N 40033,O=C1NCC2CN(C(c3ccccc3OC(F)(F)F)=O)CC12 40034,c1(NC(CC2C(CNC(CCSC)=O)C2)=O)cnc2[nH]cnc2c1 40035,Cc1ccc([N+](=O)[O-])c(C)c1C(N1CCC1CNC(c1cnc(C2CC2)s1)=O)=O 40036,N1(C(c2noc(CC)c2C)=O)CC(NC(c2ccc(C#N)[nH]2)=O)CC(O)C1 40037,C12(C(=O)OC)CCOCC1CN(C(=O)Cc1ccccc1OC(F)F)C2 40038,c1(NC(C2CC(O)CN2C(c2ccc(S)cc2)=O)=O)cccc(C(F)(F)F)c1 40039,C1(C(=O)NCC2(C)CCCC2O)C2CCC(C2)C1NC(C1(C)COCCO1)=O 40040,c1(OCC(=O)NCC2CC(NC(Cn3c(C)ccn3)=O)C2)ccccc1Br 40041,Cc1ccccc1C1(C(N2CCC(NC(C3CC(OC(F)F)C3)=O)C2)=O)CC1 40042,c1(CNC(C2C(OC)CCC2)=O)ccc(CNC(c2c[nH]c(C)c2)=O)cc1 40043,C1(NC(CSc2c(C)cccc2)=O)CN(C(=O)CCCC(C)N(C)C)CC1(C)C 40044,CC(CC(=O)N1CC(F)(C(N2CCCC(NC(N)=O)C2)=O)C1)C(F)(F)F 40045,c1(C(N2CC(CNC(C(c3ccccc3)OC)=O)C2)=O)c2c(nn1C)CCSC2 40046,c1(C(=O)NC(C)CCCNC(c2csc(=N)[nH]2)=O)nccn2nccc12 40047,N1(C(c2cc(C)on2)=O)CC(C)(C)OC2(C1)CN(C(C1C3(CC3)C13CC3)=O)C2 40048,CC1=NS(=O)(=O)NC=C1C(=O)N1CC(NC(c2c[nH]cc2C)=O)CCC1C 40049,C1(N(C(COCC#C)=O)C)CN(C(C2CCCCN2S(C)(=O)=O)=O)CC1(C)C 40050,O=S(=O)(c1ccc(Br)cc1NCC1CCCC(O)C1)NCC(C1CC(C)(C)C1)O 40051,CCCC(CC(C)C)C(=O)N1CC(COC)(NC(=O)CCC(=O)NCCC)C1 40052,C(=O)(CCC(C)(F)F)NC1C(OC)CN(C(=O)CC2CCCCC2)C1 40053,N1(C(C(C2CCCCC2)C)=O)CCCC2(NC(c3nc(=O)n(C)[nH]3)=O)CCCC12 40054,CCCCCC(C)(CC)C(=O)N1CC2CCC(C1)N2c1ccncn1 40055,c1(C(=O)Nc2scc(C(C)NC(C3CC3C(N)=O)=O)n2)ccc(F)c(Cl)c1 40056,N1(C(=O)Nc2c(CC)nns2)CC2CC2(CNC(=O)CCN(C)CC)C1 40057,c1(C(=O)NCC(CC)NC(C2(O)CC3(CCOCC3)C2)=O)cnc2cc[nH]c2c1 40058,N1(C(CCNC(c2ccncc2)=O)=O)CCCC2CCN(C(C3(O)CC3)=O)CC12 40059,N1(C(CC2CCN(Cc3ccc(F)c(C)c3F)C2)=O)CC2CCN(C)C(=O)C2C1 40060,c1(C(=O)NCC2(F)CCC(NC(C(CCOC)C)=O)C2)cc(OC)c(O)c(N)c1 40061,N1(C(C2C(C(C)(C)C)CC2)=O)CCC2CN(C(=O)C(C)N3CCCC3)C2C1 40062,S(=O)(=O)(c1ccc(NCC2(CCO)CCOC2)c(Cl)c1)N1C(C)CC2(CCC2)C1 40063,C1(CNC(c2cn(CCC)nn2)=O)C(C)CCCN1C(C1CCC(CO)CC1)=O 40064,CCC(C)CCC(=O)NC(CO)CCCNC(=O)CCc1ncccn1 40065,c1(C(=O)NC2CC3(C(=O)NC(CO)CCCO)COC2C3)c[nH]c2ccncc12 40066,C1(NC(c2cc(COC)oc2C)=O)(CO)CCN(C(=O)C(C)CC(F)F)CC1 40067,c1(CCC(=O)N(C2CCCN(C(C3CN(C(=O)N(C)C)C3)=O)C2)C)cccnc1F 40068,N1(C(CCC2CC(OC)C2)=O)C(C(=O)NC2CCCC2CCO)C2CC(O)C1C2 40069,N1(C(CSCC(=O)OC)=O)CCC(CN(C)C(C2CSCCS2)=O)C1 40070,C(C)(C1CCCc2ccccc21)NC(=NCC)NCCc1ccc(Cl)cc1F 40071,c1(N2CC3C(NC(c4c(F)ccc(C)c4F)=O)C3C2)ncnc2sc(C)nc12 40072,C1(C(N2CC(NC(C3CC4(CCCC4)CO3)=O)C2)=O)C2Cc3ccccc3C12 40073,CCCCC(CNC(=O)CCOCC)NC(C1C=C(C)CS1)=O 40074,c1(Cc2cn(C3CCN(C(C(=O)N(CC)CC)=O)C3)nn2)ccc(Br)cc1F 40075,c1(C(C(N2CCCC(N(C(CC(=C)C)=O)CCO)C2)=O)C)c[nH]c2ccccc12 40076,C(CC(C)C)(C(=O)N1CCCC(CNC(c2c(C)noc2C)=O)C1)OC 40077,n1(CC(C)C)cccc(C(=O)NCC(C2CC2)NC(=O)C(O)CN(C)C)c1=O 40078,C=C(C)C(O)CC(=O)NCCC1CN(C(c2cnn(CC3CCOC3)c2)=O)C1 40079,C12(CC(=O)NC3(C(C)C)CC3)CCC1CN(C(C1CCCCNC1=O)=O)C2 40080,CC(C)C(O)C(C)(C)C(=O)NC1C=CC(C(=O)NCCC(C)C(F)(F)F)C1 40081,C(C(C)C)(C(O)C(=O)N1CCCCCC1C(=O)N(C(C)CC1CC1)C)OC 40082,C(=O)(C#CC1CCCOC1)N1CC2C(NC(c3ccc(F)s3)=O)C2C1 40083,N1(C(CCSC)=O)CCC2(C1)C(=O)N2.C1(CO)(CO)CCC1 40084,C1(NC(c2ccc(C)nc2)=O)CN(C(c2ccc(SC(F)(F)F)s2)=O)CCC1C 40085,C=CCC(C)(C(F)F)NC(=O)CC(C)CNC(c1ccncc1OC)=O 40086,Cc1nc(C)c(CC(=O)NCCCC2(NC(=O)CN(C)CCO)CC2)c(O)n1 40087,CCCC(C(=O)NCCCCCN1CCN(C(C2COC(=O)C2)=O)CC1)N(C)C 40088,C1(CNC(c2cc(C)on2)=O)(CO)CCN(C(=O)CC2CCCC2C)CC1 40089,C1(C(=O)NCC(C)(C)NC(c2ncoc2Br)=O)CCOCC1(C)C 40090,C(=O)(C(F)CC(C)(C)C)N1C(C(=O)NC(c2c(C)nccn2)C)COCC1 40091,c1(C(=O)NCCCN(C(C(C)C2CCCC2)=O)C)cc(F)cc(S(N)(=O)=O)c1 40092,C(CCC(C)CC(=O)N1CC(O)(CCNC(C2CCCOC2)=O)C1)=C(C)C 40093,N1(C(c2cc(C)[nH]c2)=O)C2CCC(C(=O)NCc3cncs3)C1CC2 40094,C1(CCNC(c2cc(C(=O)OC)sn2)=O)CCCN(C(=O)C(C)C2CCC2)C1 40095,c1(C(N(CC(C)NC(c2c(OC)cccn2)=O)C)=O)cc(Br)cnc1C 40096,N1(C(CC2C(C)(C)C2)=O)CCCCC12CN(C(C1SC3C=CC1CC3)=O)C2 40097,C1(CC(C)NCC(O)Cc2ccccc2)CCC(=O)N1 40098,C1(OC)(CO)CCN(C(C2CCC=CCC2)C(=O)NCCCSCN(C)C)C1 40099,C1(CNC(C2C(CCC)C2)=O)CN(C(=O)Cc2c(C)cccc2Cl)C(C)(C)C1 40100,CS(=O)(=O)c1cc(C(N2CCC3CN(S(=O)(=O)CC4CC4)CCC23)=O)ccc1F 40101,C1(NC(C(c2n(C)ncc2)O)=O)(COC)CCN(C(=O)CSc2nncn2C)C1 40102,Cc1cc(Cl)c(C(N2CC(C)(C)C2Cn2cc(C3CCCCO3)nn2)=O)s1 40103,C1(N(CC(N2CCCCC2)=O)C(=O)NC2CC(CC)C2)CCS(=O)(=O)C1 40104,C(=O)(C1=NOC(C)C1)NCCN(C(C1C(C=C)OCC1)=O)C 40105,C1(NC(CC(=O)OC)=O)CC(O)CN(C(=O)Cc2ccc(OC(F)(F)F)cc2)C1 40106,C(CCCCC(=O)N1CC2CC1(CNC(=O)Cc1cc(C)cs1)C2)OCC 40107,c1(C(=O)NC2CCCN(C(C3C4COCC34)=O)C2)cc2oc(Br)cc2s1 40108,c1(CC(=O)NC2(COC)CN(C(c3cc(C#N)cs3)=O)C2)cnccc1Cl 40109,C(=O)(C(CC)n1cccn1)NCCNC(C=C(CC)C)=O 40110,C1(CC)CCCN(C(=O)CC2CC(F)C2)C1C(=O)NCCCCc1ncc[nH]1 40111,c1(CCOc2ccc(C(=O)OC)c(F)c2)csc2sc(C)cc12 40112,O=S(=O)(c1cccnc1NCCC1CCC2CC12)NCc1cc(C(F)F)on1 40113,c1(C(=O)NC2C(C)N(C(=O)CCc3cnoc3)CC2)nccc2[nH]ccc12 40114,Cc1c(C(N2CCN(C(=O)C(C)(C)CO)CC2CS(C)(=O)=O)=O)cccc1C#N 40115,C(C(CC(C)C)C(=O)NC1CC(CCNC(=O)C(C2CCCC2)OC)C1)OC 40116,C(C(C)(F)F)N(C(C=CC(C)NC(C1(C(N)=O)CC1)=O)=O)C 40117,N1(C(C2CCSCC2)=O)CC2CCC(C(N3CCC(N4CCCC4)C3)=O)(C2)C1 40118,c1(C(C(=O)NCCOCC)N(C2(CCO)CC2)C)ccc(C2CCC2)cc1 40119,N1(CC(N2CCCN(C(CCC#CC)=O)C(C)C2)=O)CCSC2CCCCC12 40120,C1(C(N(Cc2cn(-c3c(C)cc(Cl)cc3)nn2)O)=O)C2CCCC1CCC2 40121,N1(C(c2cccc(CC)c2)=O)CCC2(CC1)CC2NC(C1(C)CCSCC1)=O 40122,N1(C(c2ccc(OC)s2)=O)CCC2CN(C(c3cc(N)cc(O)c3)=O)CC12 40123,CC1OC2(CO)CC1(C(N1CC3CC1CN3C(=O)C(F)CC1CC1)=O)C2 40124,C1(C(F)F)(CNC(CC(=O)NCC)=O)CCN(C(c2cnn(C)c2OC)=O)C1 40125,c1(CC)nc[nH]c1C(N1CCCC1CN(C(=O)CC1CCSCC1)C)=O 40126,C1(C)(C(=O)NCCC(C)N(C(=O)CCCCN2CCOCC2)C)CCC12CCC2 40127,c1(C(=O)NCCOCCN(C(CC2CCCC(OC)C2)=O)C)cc(Cl)ccc1N 40128,C1(C(N2CC(OCC(=O)NCc3ccc[nH]3)C2)=O)Cc2nccn2C1 40129,N1(C(c2cnn(CCC)c2C)=O)CC2CC(C1)N(C(=O)CCC(C)C#N)C2 40130,C1(NC(Cc2cnc(C)s2)=O)CC(N=c2[nH]c3cccc(F)c3s2)C1 40131,C1(N(C(C(C)OCC(F)(F)F)=O)C)CN(C(=O)CCc2nccs2)CC1(C)C 40132,c1(C2C(C(=O)NCCN(C(=O)Cc3cnn(C(F)F)c3)CC)C2)ccccc1Cl 40133,C1(NC(C(C)CNC(c2ccccc2)=O)=O)CN2CCC1(F)CC2 40134,c1(C(N2C(CNC(C3C(C=C)CC3)=O)CC(C)(C)C2)=O)ccc(Cl)c(N)c1Cl 40135,N1(C(c2c(C)nsc2C)=O)CC(NC(=O)CC(O)CN(C)C)CC2(CC2)C1 40136,C(C)(CCN=c1cc(C2CCCCC2)nc[nH]1)NC(c1ccn(CC(C)C)n1)=O 40137,c1(-n2cc(C3(F)CN(C(C4(CSC)CC4)=O)C3)nn2)ccc(C)cc1C 40138,C1(C(=O)NC(COCC)C)CN(C(C2(CC)CCCC2O)=O)CC1(F)F 40139,c1(C(N(C(CNC(CC(C)OC)=O)C2CC2)C)=O)cnc2ncnn2c1C(C)C 40140,C1(CNC(CCC=CCC=C)=O)CC(NC(c2coc(Br)n2)=O)C12CCC2 40141,C1(CC#C)(C(=O)NCC(CCNC(=O)C=CCN(C)C)OC)CCOC1 40142,c1(CC(=O)NCC(C)(C)OCCNC(C(CC=C)C)=O)c(C)cc(C)nc1O 40143,CCC(C(=O)N(C)Cc1cnc(C)s1)N(C(=O)CNC(=O)NC1CC1)C 40144,N1(C(C(C(C)(C)C)NC(=O)C(F)OC(F)(F)F)=O)CC2C3CCC(O3)C2C1 40145,C(C(C(=O)N1CCN(C(C)C)C(=O)C1)C(C)(C)C)NC(CC=C)=O 40146,CN(C1CCCc2c1cnn2C)C(=O)Cc1cnn(C)c1 40147,c1(C(N)=O)cc(C(=O)NCC2OCCC2C(=O)NCC2(F)CC(O)C2)n[nH]1 40148,Cc1cc(C(N2CC3C(NC(c4cccnc4)=O)C3C2)=O)c2cc[nH]c2c1 40149,c1(OCC)cccnc1C(N1CC(CCO)(NC(=O)CCc2ccncn2)C1)=O 40150,C=C(C)CC(C(=O)NCCC1CC(F)(F)CN1C(C1CCCOC1C)=O)OC 40151,N1(C(c2n(CC)nnc2)=O)CCC(NC(=O)C(C)(C2CC2)OC)C1C 40152,c1(C(C)C)nnnn1CC(=O)NC(CNC(C1CC(F)(C(=O)O)C1)=O)C(C)C 40153,Cn1cncc1C(c1nnnn1Cc1cccs1)NCCC(=O)NO 40154,c1(C(N2C(CNC(C=CC(N)=O)=O)CCCCC2)=O)noc2cc(F)ccc12 40155,O=C(N=c1[nH]c(Cl)ncc1O)C1CN(S(=O)(=O)C2CC2)CCC1O 40156,C1(N=[N+]=[N-])(C(=O)NC(C(C(=O)OC)C)C)CCN(C(C2CCCC2C(C)C)=O)C1 40157,N1(C(CC(C)N2CCCC2=O)=O)CCC(C(F)F)(CNC(C2(Cl)CC2)=O)C1 40158,c1(C(=O)NCC2CCN2OC)cccn2nncc12.c12csc(c1)C(=O)NC2 40159,C#CC1CCN(C(=O)C(CCC=C)NC(C2CCS2(=O)=O)=O)CC1 40160,c1(C(=O)NC2CCN(C(CC(C)C(F)(F)F)=O)C(C)C2)c(N)c(F)cc(F)c1F 40161,CCC(Cc1ccccc1)C(=O)NC(C)CNC(c1cc(C(F)(F)F)no1)=O 40162,S(=O)(=O)(c1cc(C(=O)O)c(Cl)cc1Cl)N1C(C(=O)O)CCC(C(F)(F)F)C1 40163,Cc1cc(-n2cccn2)ccc1NC(C)C(C)S(C)(=O)=O 40164,C=C(C)C(C)(C)C(=O)NC(C1CCN(C(C2CCC(C(=O)OC)O2)=O)C1)C 40165,c1(C(N2CCC(O)(C(C)NC(=O)C(O)C3CCCC3)C2)=O)ncc2ccccn12 40166,C(=O)(NN1CCCC1C(N1CC(O)(C(F)(F)F)C1)=O)C1(CC(C)=O)CC1 40167,N1(C(CC(C)(C)OC)=O)CCC(CO)C(NC(=O)C(C)(C)c2csc(C3CC3)n2)C1 40168,c1(C(=O)NCCC2CN(C(C=C(COC)C)=O)C2)cc(C)c(C)c2ncccc12 40169,N1(C(C2CCC(N(C)C)CC2)C(=O)NCCC(=O)OCC)CCCOC(C)C1 40170,N1(C(CCC2(C)N=N2)=O)CCC(CCC(=O)NCCc2cnnn2C)C1 40171,S(=O)(=O)(c1cnc(NC(c2cccc(Cl)c2C)C)c(Cl)c1)NC(COC)C1CC1 40172,n1(CC)nc(C)c(C(=O)N(C)CC2CCN(C(=O)CC(C)OC)C2)c1Cl 40173,C1(Cl)(C(=O)OCC)CC12CCN(Cc1cnn(Cc3ccncc3)c1)CC2 40174,CCC(O)C(C)C(=O)N1CC(C(F)Cn2cc(-c3ccc(C)cc3C)nn2)C1 40175,C(=O)(C(O)CCCNC(=O)C=CC(=O)N(C)C)NCCC(CC)C 40176,C(C(CNC(=O)CCc1cnoc1)NC(=O)CC1CC(C(C)(C)C)C1)OC 40177,CC1(C)C(NC(c2cc(C3CC3)no2)=O)CCN1C(=O)Cc1cnoc1 40178,C=CC(CCC)CC(=O)NC(CC1CC1)C(=O)NOCC(O)C(C)(C)C 40179,N1(C(CNC(CC)=O)=O)CC2CCC1C1CN(C(=O)Cc3ccsc3)CC21 40180,C(=O)(CCN(OC)C(=O)C(C)(O)C(F)(F)F)NCC(C#C)CC 40181,C1(S(C)(=O)=O)(C(N2CCCC(NC(C=CCOC)=O)(CO)C2)=O)CC(O)C1 40182,C1(NC(C2Cc3n(cc(C)n3)C2)=O)CC2CCC(C1F)N2C(C1(C)CC1(F)F)=O 40183,N1(C(c2ncn(C)n2)=O)CCOCC(CNC(=O)CC(C2CC2)C2CC2)C1 40184,C(=O)(C(O)CC(C)C)N(C1CN(C(c2c(C)cc(F)s2)=O)CC1O)C 40185,c1(CC(=O)N(CC(C)NC(=O)COC2CC(F)(F)C2)CC)cccc(OC)c1F 40186,N1(C(CC(C)n2cccc2)=O)CCC(NC(C2CCCN2N=O)=O)C12CCC2 40187,N1(C(CCOc2ccc(C)cc2)=O)CCN(C(C2CCCCN2C)=O)CC1C 40188,c1(C(=O)NCC2CCCC(C)C2)cccc(S(C)=O)c1 40189,c1(-n2c(C(c3cnn(C)c3)C)nc(C(C3CC3)OC)n2)ccc2c(c1)OCCO2 40190,c1(C(=O)NC(C(C)NC(c2c(CCC)nco2)=O)CO)cc2cccc(C)n2n1 40191,CC1CN(C(C)C(=O)N(CC(=O)NC(C(N)=O)C2CCCC2)C2CC2)C1 40192,C1(NC(c2csc(-c3ccco3)n2)=O)CC(O)CN(C(C2CC(O)C2)=O)C1 40193,C(C(CC(=O)N1CCC(CO)C1)N(C)C)NC(CN(C(COC)=O)C)=O 40194,C(=O)(CCC(=O)NN(C)C)N(C(C)(C)C(C)CC(=O)N1CC(CC23CC(C2)C3)C1)C 40195,c1(CC(=O)NC2CCC(NC(C3C(C(N)=O)C3)=O)CC2)cc(Br)ccc1Cl 40196,c1(-c2n(-c3cccc(OC)c3Cl)nc(CO)n2)cc(C2CCCO2)c(C)nc1O 40197,C1(CC)CN(C(=O)C=C(C)c2cccs2)CC1NC(C1(C(C)(F)F)CC1)=O 40198,c1(OC)cc(N)c(Cl)cc1C(=O)NCC1(NC(C2CC23CC(O)C3)=O)CCOC1 40199,CC1(O)CCN(C(=O)C(c2cn(C)nn2)NC(C2(F)CCCCC2)=O)CC1 40200,N1(C(c2c(C)c(F)ccc2)=O)CCC2CCCN(C(c3cnco3)=O)C2C1 40201,C1(C(=O)NC(C)CN=[N+]=[N-])CN(C(C2CC(=C3CCC3)C2)=O)CCC1(C)C 40202,c1(C(c2n(CC=C)nnn2)NCC2(n3cccn3)CC2)cc(Cl)cc(C)c1OC 40203,c1(CN(C(Cc2cc(C)no2)=O)C)cccc(CNC(C2CCCC(O)C2)=O)c1 40204,C1(NC(COCCCOC)=O)CC12CCN(C(c1cncc(OC(C)C)c1)=O)C2 40205,N1(C(c2c(C(N)=O)cccc2)=O)CCC(F)C(NC(C2CCC(F)CC2)=O)C1 40206,c1(NC(C2(F)CN(C(c3c(C(C)C)cccc3)=O)C2)=O)cc([N+](=O)[O-])ccc1I 40207,CC1OCCC1(F)C(=O)NC1CC(C(=O)N(C)CCC2CCCCC2)C1 40208,C12(CCNC(COCC#C)=O)CCC(C1)N(C(=O)C=C(C)C(C)C)C2 40209,c1(C(N2CCC(C(C)NC(c3ccc(C4CC4)o3)=O)C2)=O)cc2c(s1)CCCC2 40210,C1(=O)C(CCC(N)=O)n2cc(nn2)N1CC=C.C1(CC2(O)COC2)CCC1=O 40211,n1(CC)nccc1CN(C(=O)CN(C(=O)CNC(=O)NCCOC)C)C 40212,C1(C2CCCCO2)(C(=O)NCC(CNC(c2c(CC)cno2)=O)(C)C)CCCO1 40213,C1(C(N(C(=O)CN2CCOCC(O)C2)C2CC2)=O)CC2(CCC2)CO1 40214,C1(NC(C(C(C)C)C)=O)CC2(COC(C)C2)C1 40215,N1(C(c2c(C)onc2)=O)CCN(C(C2C(C)C2C)=O)C2(CCC2)C1 40216,c1(CC(=O)NC(CCNC(CCCOCC)=O)C)cccc(Br)c1 40217,c1(C(=O)NC2CCC(N(C(=O)OC)C)CC2)ccc(C(C)=O)nc1O 40218,C(=O)(C(O)CC[S+](C)C)NCC1(F)CCN(C(C2(COC)CC2)=O)C1 40219,c1(C(N2CCN(C(c3cnsn3)=O)C(C3CCC3)C2)=O)nccc2[nH]ccc12 40220,[N-]=[N+]=NCCC(=O)NCCC(O)C(=O)N1CCOC(C2CCC2)C1 40221,C(=O)(C(F)C(CC)CC)N1C(CNC(CSCCCC)=O)CC(OC)C1 40222,N1(C(=O)CCCc2cncs2)CC2(CCCCN2C(=O)CCN2CCOCC2)C1 40223,Cc1ncc(C#N)cc1NC(=O)C(C)CN(C(=O)CC1OCCC1(C)C)C 40224,C(CN=c1ccnc(NC2CC(C(C)(C)C)C2)[nH]1)N1CCCC(C)C1 40225,c1(C(=O)NC(CCNC(Cc2ccn(CC)n2)=O)C)cc(C)cc(O)c1 40226,c1(C(=O)NC2CC(C)(C)CN(C(=O)C#CC3CC3)C2)c[nH]c2ccncc2c1=O 40227,C1(NC(CCNC(CC(C)C)=O)=O)CN(C(=O)C(C)(C)C(F)F)CCC1O 40228,CC(C)C(CC(F)(F)F)OC(=O)CCC#CCc1ccccc1 40229,c1(-c2nnc(C(COc3c(C)cccc3)OC)n2C)c[nH]c2cc(C#N)ccc12 40230,N1(C(C(C(C)C)CO)=O)CC=C(CCNC(c2cc(F)c(CO)c(F)c2)=O)CC1 40231,c1(C(=O)NCC(CC=C)NC(CCC#C)=O)ccc(OC(C)C)nn1 40232,C1(C(N(C(CCNC(c2c(C)ncnc2)=O)C)C)=O)COc2ccc(F)cc2C1 40233,c1(NC2CC(C)N(C(=O)CCCc3ccsc3)C2)ncc([N+](=O)[O-])cc1Cl 40234,O=C1CN(CC(=O)NCc2nc(CNC(C3(C4CCC4)CC3)=O)cs2)C(=O)N1 40235,c1(C(=O)NC2C(CNC(=O)CCOC3CCOC3)C2)c(Cl)ccc2ncccc12 40236,c1(C(N2C(C3(NC(=O)C=C(Cl)Cl)CC3)CCCC2)=O)cccn2cncc12 40237,C12(NC(CCc3ccc(C)o3)=O)CCN(C(c3csnc3Br)=O)CC1C2 40238,C(=O)(CC(C(C)OC)NC(C1CCOC1)=O)N(C(CC)CO)C1CC1 40239,C(C(=O)NCC=C(C)C)(C1(C)CC1)NC(C=CC=CC)=O 40240,c1(C(N(C(C)CCNC(=O)CC2CCC(F)(F)C2)C)=O)cccc2c1CCC2=O 40241,C(C(CO)C(F)(F)F)NC(C(C)CNC(C1CC1(F)Cl)=O)=O 40242,C#Cc1c[nH]nc1C(N1C(C(N2CC(C(CC)CC)C2)=O)CC1C)=O 40243,C1(NC(C2(COC)CCCC2)=O)COCCN(C(=O)Cn2cc(Cl)cn2)C1 40244,C(=O)(C1=CCCCO1)NC(COC)C(=O)NCC1CC(=O)NC(C)C1 40245,C1(CNC(c2cnc(CC)s2)=O)(OC)CCN(C(=O)C(F)(F)c2nccs2)C1 40246,c1(C(=O)NC2CC(NC(C=NOC)=O)C2)cnc(O)c2c1NCCC2 40247,c1(OC)ccc(Cl)cc1CC(=O)NCC(C)(C1CC1)NC(=O)CCc1ccsc1 40248,N1(C(c2nc(CNC(C(C)C3CCCC3)=O)oc2)=O)CC(C2CCCCC2)C1 40249,C12(C(=O)NC3CCCN(C(c4c(CC)c[nH]n4)=O)CC3)CC3CC(CC1C3)C2 40250,C12(NC(C(=O)NC(c3ccc(F)cc3Cl)(C)C)=O)CCC(CO)(C1)OC2 40251,C(CCC)(C(=O)NCCC1(NC(=O)COc2ccsc2)CCCC1)=CCC 40252,C1(C(=O)NC2CC(NC(CC(C=C)(C)C)=O)C2)COc2ccc(OC)cc2C1 40253,Cc1nc(=N)[nH]cc1C(N1CCN(C(=O)Cn2ccnn2)CC1C1CC1)=O 40254,C1(C(=O)NCCC(C)NC(=O)C(c2ccc(F)cc2)(F)F)CCCCN1C 40255,C1(C(=O)NC(CC)C(=O)NC)CNC(=O)CN1C(=O)C1=COCCC1 40256,c1(COC)nc(NC2CN(C(c3ccn(C)n3)=O)CCC2C(F)(F)F)cc(O)n1 40257,Cc1nn(C)cc1C(O)C(=O)NCc1cccc(NC(c2coc(O)n2)=O)c1 40258,c1(C(=O)Nc2ccnc(N3CCOC(C(F)(F)F)C3)c2)cc2c(cc1O)CCCC2 40259,CC(C)CC(O)C(=O)NC(C)CNC(c1cc(C(F)(F)F)cc(N)c1)=O 40260,C(=O)(C1CCCn2ccnc21)NCC1N(C(C2N(CCCC)CCOC2)=O)CC1 40261,N1(C(C=CCNC(C2CC(C)(O)C2)=O)=O)CCc2ncccc2C1 40262,C12(C=CCN1C(=O)COCCCN=[N+]=[N-])C(=O)NC2.C1(SC)CC(N(C)C)C1 40263,C(c1ccc(F)c(F)c1)=C(C)C(=O)NC1CN(C(c2nc(Cl)c(Cl)s2)=O)CC1C 40264,c1(NC(CNC(=O)NCCc2nn(CC)c(C)c2)=O)ccc2ncsc2c1Br 40265,N#Cc1cncnc1N1CCCC(NC(c2ccccc2O)=O)C1 40266,N1(C(c2nc(CC)sc2)=O)CC(NC(=O)C(c2ccccc2OC)(C)C)CC1C 40267,C12(C(C)C)CC1CN(C(=O)CC(C)NC(C1CCCCC1O)=O)C2 40268,c1(C(=O)NC(C2CN(C(C(=O)NCC)=O)C2)C)ccc2nnc(O)n2c1 40269,c1(C(=O)NC(CCOCC)C(=O)N2CC(c3nn[nH]n3)C2)cccc(=O)n1C 40270,c1(CC(N2CC(C)N(C(C3CC(OC(F)F)C3)=O)CC2)=O)cccc([N+](=O)[O-])c1 40271,Cc1ccc(C(=O)NC2CCCCC2c2ccccc2F)cc1N1CCOCC1 40272,O=C(C(O)Cn1cncn1)NC1CN(C(C2CC2(Cl)Cl)=O)C1 40273,Cc1nc(CO)sc1C(=O)NC1CN(C(c2ccccc2CO)=O)C1.C1(C(C)C)CC1 40274,c1(-c2cn(C3(C(=O)NCC(=O)NCC)CCCC3)nn2)ncccc1C(F)(F)F 40275,C1(C(=O)NCC2C(CNC(CC=CC)=O)C2)CCc2ncsc2C1 40276,c1(C(=O)NC(C)CC(C)NC(=O)Cc2ccc(C#N)cc2)cnc2[nH]ccc2n1 40277,Cn1nc2nc1S2.C1(NCC(=O)NC(=O)C2CC2)CCCCC1 40278,N1(C(c2cnc(C)s2)=O)CCC(NC(c2cc(=O)n(C)o2)=O)CC1C 40279,C1(C(=O)NCCc2ccc(CC(C)C)cc2)CCCC12CCN(C(=O)C(C)C)C2 40280,c1(C(=O)NC23CN(C(C4(OCC)CCCC4)=O)C(C2)C3)ccc2n[nH]cc2c1 40281,c1(C(=O)NCCCN(C(CC(C)n2ccnc2)=O)C)cccc(P(C)(C)=O)c1 40282,c1(CC(=O)NC2CC(O)(CNC(CCN(C)CC)=O)C2)ccc(S(C)=O)cc1 40283,Cc1ccsc1-c1cn(C(C)C(=O)N(C2CC2)C2CC2)nn1 40284,CCCC(CC(C)C)C(=O)NCC1(F)CC(CNC(c2cc(N)ccn2)=O)C1 40285,NS(=O)(=O)C1CN(C(=O)Cn2nnc(-c3ccc(Cl)cc3)n2)C2(CCC2)C1 40286,c1(CC(=O)NCc2c(CCNC(C(C)(C)C3CC3)=O)ocn2)ccc2c(c1)CC2 40287,c1(C(N2CC3C(CNC(C(CCC)N(C)C)=O)C3C2)=O)cn(C)c(C)cc1=O 40288,CC1(C)C(C(=O)NC(CCO)C2CC2)CCN1C(=O)CCCn1cccn1 40289,Cc1nc(C(C)C)ncc1C(=O)NCCCN(C(=O)CNC(c1ccco1)=O)C 40290,CC(CNC(C1COCCC1C)=O)C(F)C(=O)NC1(CC2CCC2)CC1 40291,n1(CC=C)c(SCC2NCCC2C)nc2sc3c(c2c1=O)CCC3 40292,C=CCC(F)(F)C(=O)NCC1(C)CCC(NC(=O)CCSCC)C1 40293,N1(C(C=C(C)Cl)=O)CCCN(C(=O)CCOC2CCC2)C(c2ccccc2)C1 40294,CC(C)C(O)C(F)(F)C(=O)NCC1C(C)CCCN1C(=O)CCc1cnc[nH]1 40295,c1(C(=O)NC(CNC(C2C(=C)CC2)=O)CCOC)c(C)cc(C)oc1=O 40296,C1(C(N2CC(OC)CC2(C)CNC(=O)CS(C)(=O)=O)=O)CC2(C1)CC(C)(C)C2 40297,C1(N(C(CNC(CC)=O)=O)C)CCN(CCSc2cc(C)c(C)s2)CC1 40298,CCCCCC(C)CC(=O)NCCC(O)CNC(c1ncoc1C1CC1)=O 40299,CC(C)CC(C(=O)N(C)CC1(CO)CC1)NC(C1CCC(=O)N(C)C1)=O 40300,C(CCSC)(C(=O)NCc1cn(CCNC(=O)CCc2ccccn2)nn1)OC 40301,C1(C(=O)NC(CCCOC)(C)C)CCC(O)CN1C(=O)CCCn1cccc1 40302,C1(C(N2CCC(F)C2)=O)CC2OCCC2N(C(C2Cc3ccccc3C2)=O)C1 40303,c1(C(=O)NC2C(NC(=O)C=Cc3cocn3)C2)cc2c(s1)CCCC2 40304,Cc1nn(C2CCC2)cc1C(N1CC(CNC(=O)CCC(=O)C2CC2)C(O)C1)=O 40305,CCCC(CCC)C(=O)Nc1cccc(C(N2CCCC2C(N)=O)=O)c1 40306,Cc1nc(N2CC3CC3(C(=O)Nc3nc4c(s3)CCC4)C2)c2c(n1)CCC2 40307,Cc1cc2sc(C(=O)N(CCC(C(C)(C)C)NC(C3(C)CC3(F)F)=O)C)cc2s1 40308,C(=O)(C(C)(C)C(C)(F)F)N(CCNC(C1CC1C1(O)CCC1)=O)CC 40309,N1(C(CCOCCC)=O)CCC(CN2CCN(C(c3cscc3C)=O)CC2)CC1 40310,c1(CCNC(C(=O)NC2CC(C)SC2)=O)ncccc1N1CCCC1 40311,N1(C(C(CC2CCOC2)NC(=O)OC(C)(C)C)=O)CC2(CNC(=O)OC2)C1 40312,C1(CNC(C(CC)COC)=O)(OC)CCCN(C(C2(c3ccncc3)CC2)=O)C1 40313,c1(C(=O)NCCC2CC(NC(C3CC3Cl)=O)C2)cc2c[nH]cnc-2n1 40314,Cc1ccc(F)c(C(N2CCCC(C)(CNC(c3c[nH]c(C#N)c3)=O)C2)=O)c1F 40315,O=C1CCC2(C(=O)NCC3(O)CCN(C(c4cnsc4)=O)CC3)CCCCC2N1 40316,C1(OC)CN(C(c2c(C)noc2N)=O)CC1C(N1CC2CCC1C2)=O 40317,N1(C(c2cc(C)n(C(C)(C)C)n2)=O)CC(NC(=O)CN2CCC(C)C2)CC(F)C1 40318,c1(C(N(C2CCCN(C(c3csnc3Cl)=O)C2)CCO)=O)ccc2[nH]ccc2c1 40319,c1(C(C)NC(c2nnn(-c3ccccc3)c2C(F)(F)F)=O)c(F)cccc1F 40320,n1(CC)ncc(C(N2CCN(C(=O)CNC(=O)C(C)OC)CC2)=O)c1C(F)(F)F 40321,N1(C(C2(C)CCCC2)=O)CCCC(O)(CNC(c2cc(C3CC3)nnc2O)=O)C1 40322,N1(C(C(C)=CC2CC2)=O)CCC2CC2(C(=O)Nc2cccc(CO)c2)CC1 40323,CC(CCNC(=O)C=Cc1ccco1)CCNC(C1COCCN1C)=O 40324,c1(C(N2CC(C(C)NC(c3c(C)scc3)=O)C2)=O)cnc2ccccn12 40325,C1(OC2(CC(=O)N(CC(=O)OC(C)(C)C)C)CCC2)CCCCCC1 40326,c1(C(N2C3C(CNC(CC=CC=C)=O)C(CCC3)C2)=O)nc2n(c1Cl)CCCC2 40327,N1(C(C(C)=CC)=O)CCc2nc(CNC(C3(C(F)(F)F)CC=CCO3)=O)sc2C1 40328,C=C(C)CCCC(=O)NCC(CCOC)NC(c1nc(OC)cc(OC)n1)=O 40329,c1(C(C)C)ccc(C2CCCN(C(=O)C(C(C)O)N3CCNCC3)C2)cc1 40330,C12(CC(=O)N(c3ccc(CO)cc3)C)CCC1CN(C(c1ccncc1N)=O)C2 40331,C(=O)(C(C#N)CC)N1C(CCC(=O)N(CCN2CCOCC2)CC)CC1 40332,C1(CC=C)(Nc2cccc3cncn23)CC2CCC(C1)N2C(=O)OC(C)(C)C 40333,c1(-c2ccc(C(F)F)cn2)cc(F)ccc1F 40334,CC(C)(C)CC(C)(C)C(=O)NCC1CCN1C(c1ccc(O)c(Cl)n1)=O 40335,C1(O)(C(=O)Nc2cn[nH]c2)CC(C)(C)C1.C12COCCC1C(=O)N(C)CC(=O)N2 40336,N1(C(CC2CN(C)C2)=O)CC(NC(=O)CCNC(c2ccoc2)=O)CC(F)C1 40337,c1(CCNCc2cc(C)n(C)n2)ccc2ccccc2c1.C1(C)C(=O)N1 40338,c1(N(CCC)C)ccc(C(=O)NC23CC2CN(C(=O)C(C)n2cccc2)C3)cc1 40339,CCC(C)C(O)CC(=O)NCC(C)(C)OCCNC(c1cnc2ccccn12)=O 40340,C1(NCc2cn(CCC(=O)N(C3CCN(CC)CC3)C)nn2)CCCC(C)(C)C1 40341,c1(CC(=O)N(C)CC2(NC(c3nocc3Cl)=O)CC2)ccc(Cl)c(Cl)c1 40342,N1(C(COCCCCC)=O)CCC(CCC(=O)NCc2scnc2C)C1 40343,c1(C(N2CC(CC(C)NC(CC=C(C)C)=O)C2)=O)csc(C2CCCO2)n1 40344,Cn1ccc2cccc(C(N3CCC(C)(NC(C4CCCSC4)=O)C3)=O)c12 40345,N1(C(C2C(C)=C2)=O)CC2CCC(C1)N2C1CCN(C(=O)C(C)(C)C(F)F)CC1 40346,c1(C(C(=O)NC2CCCC2)N(CC(C)C)CCC#N)cnc2n1CCC2 40347,N1(C(CCCCSC)=O)CC2=C(C1)CN(C(c1cnc(C(F)F)c(C)c1)=O)C2 40348,c1(C(N(C2CN(C(C(CC)(F)F)=O)CC2O)C)=O)cc(F)c(C(C)C)cc1F 40349,c1(C(=O)NCCC2(C(=O)NCC3CN(C)C3)CC2)ccc2nccn2c1 40350,c1(C(=O)NCC(C)N(C(=O)Cc2cc(Cl)ccc2O)C)cccc2c[nH]nc12 40351,C(=O)(C1=CCC(C)(C)CC1)NCC1(F)CCCN(C(CSCC=C)=O)C1 40352,c1(OC)cc(C(=O)NCC2CN(C(C3CC3(C)C(C)C)=O)C2)c(C)c(Br)c1 40353,C(CC(C)C(=O)N1CCC(CN(C)C(c2cncc(-n3cccn3)n2)=O)C1)=CC 40354,CC(C)C(CC(=O)NC1CCCCNC1=O)NC(C1CC(N=[N+]=[N-])C1)=O 40355,C(=O)(CN1C(=O)CCc2ccccc21)NCC1C(NC(CC2CN(C)C2)=O)CC1 40356,c1(NC(CC(CC)C)=O)ccc(Br)cc1F.C12CCN(CC1)CC=CC(=O)N2 40357,CC1(C)COCCC1C(=O)NC1C2CCN(C(c3ccc(F)cn3)=O)C12 40358,C1(CNC(=O)NCCN(CCC)C)CCC1C(=O)OCC 40359,N1(C(Cc2c(C)cnn2C)=O)CCN(C(=O)COc2ccsn2)CC(O)C1 40360,C(=O)(C(C)C(C)NC(C1(COCC)CC1)=O)NCC1CCOC1 40361,c1(C(=O)NCCC2(O)CN(C(C3C(C)CC3C)=O)C2)ccnc2ncnn12 40362,N1(C(C(C)(C)F)=O)CCC2(CCN(C(c3coc(-c4ccc(F)cc4)n3)=O)C2)C1 40363,N1(C(C2C(C)(C)CCN(C(C3CCCC3F)=O)C2)=O)CCC2(CCCCO2)C1 40364,c1(C(=O)NC2CC(CS(N)(=O)=O)C2)cccc(C(=O)O)c1 40365,Cc1ncc(C(=O)NCC2(C(=O)NC(C)(CO)C(F)(F)F)CC2)c(C)n1 40366,C1(NC(c2c(C(C)C)onc2)=O)CC(C)N(C(c2cn(C)cn2)=O)C1 40367,N1(C(COCCOC)=O)CCN(C)C(CNC(C2CN(C)CCO2)=O)C1 40368,C1(NC(C2(C)CCC2)=O)CCC2(CC1)CCN(C(=O)CC1CCCC1(F)F)CC2 40369,C1(CNC(=O)C2=C(Cl)CC2)CCN(C(=O)CCF)CCC1(F)F 40370,Cc1csc2ncnc(NC(C)CC(C)NC(c3ccc4nccnc4c3)=O)c12 40371,c1(C(N2CC=C(CNC(=O)C=CC3CCC3)CC2)=O)ccc2c(c1)C(=O)NC2=O 40372,c1(CC)nc(N2CCCC(NC(c3sc(CC)nc3C)=O)C2)c(CC)c(Cl)n1 40373,O=C1Cc2cc(C(=O)NC3CN(C(C4CS(=O)(=O)C4)=O)CC3O)ccc2N1 40374,c1(N2CCCC(NC(=O)C=Cc3ccc(Br)s3)CC2)cc2ncnn2cn1 40375,c1(C(N(CCOCCN(C(C(C=C)CC)=O)C)C)=O)ccc2c(c1)OCC2 40376,Cc1no[nH]c1=NC(=O)C1(C)CCN(c2ncncc2I)C1 40377,c1(C(N2CC(C(=O)OC)CC(CC)C2)=O)ccc2c(Br)cnn2c1 40378,N1(C(C(C=C)OC)=O)CC(CC(=O)NCC(C)(O)CCC)C2(CC2)C1 40379,CN1CCN(C(C2(C)CCN(C(=O)Cn3ncccc3=O)C2)=O)CC1=O 40380,C1(C(=O)NCCNC(c2ccc(C(C)C(F)(F)F)cc2)=O)CCC(N=[N+]=[N-])CC1 40381,c1(NC(CC)=O)ccc(F)c(NC(=O)CCC(=O)c2cccc(OC)c2)c1 40382,c1(C2CN(C(C=C(C)C(C)C)=O)C2)ccc(F)c(F)c1 40383,CCCCC(COC)NC(=O)CCN(C(=O)CC(OC)OC)C1CC1 40384,N1(C(C2(C(=O)NC)CC2)=O)CCN(C(c2cn(C)nn2)=O)CC(CO)C1 40385,CC1CCC(Cl)=C(C(=O)NC2CN(C(=O)CNS(N)(=O)=O)CCC2CO)C1 40386,c1(OC(C(=O)NCC(CNC(C(C)(C)OC(C)C)=O)C)C)ccc(Cl)cc1 40387,C1(C(C)C)CN(C(c2cnc(O)s2)=O)CCN1C(=O)Cc1cn[nH]c1 40388,Cc1[nH]c2ccccc2c1CNC1(c2nnnn2C2COC2)CCN(C(C)C)C1 40389,C=CC1CN(C(=O)C(CN(C)C)NC(=O)CCSCC)CCO1 40390,c1(C(N2C(C)CC(NC(C3CCC(=O)NC3)=O)C2)=O)cc(F)cnc1Cl 40391,C(=O)(CCCCC(C)CC)NC1C(CC)CN(C(=O)C(N2CCN(C)CC2)C)C1 40392,C1(CNC(c2cn(C)nc2C(C)(C)C)=O)CC2COCC2N1C(=O)C(C)(C)CO 40393,C(=O)(N=c1nn[nH]n1CCC)NC(c1ccc(Cl)cc1)CCC 40394,C(=O)(C(C)(C)C(=O)N(C)C)N1CCC(CC(C)NC(C(CC)F)=O)CC1 40395,C12(CC)COC(C(N3CC(F)(CNC(=O)Cc4ccco4)C3)=O)(C1)C2 40396,c1(CC)cc(NCC(C2CC2)N(C)C(C2CCC(CC)CC2)=O)ncn1 40397,C(C(=O)N1CCCC1C1CCCC(C)(C)C1)(C(C)(C)C)n1cc(C(=O)OC)nn1 40398,c1(C(=O)NCCOC2CN(C(Cc3cn(CC)nc3)=O)C2)csc(Cl)c1Cl 40399,c1(OC)ccc(Br)c(C(=O)NC2(c3cn(C4CCC4O)nn3)CCC2)c1F 40400,C1(CNC(c2c(C)nc(CO)o2)=O)N(C(c2cc(Cl)cn2C)=O)CCCC1(C)C 40401,c1(C(N(CC(CNC(Cc2c(C)noc2)=O)O)C)=O)cncc(-n2cccn2)n1 40402,N1(C(CC=C)=O)CCC2CCCN(C(c3cc(-c4cc[nH]n4)ccc3F)=O)C2C1 40403,C1(C2CCN(C(COCC(c3ccncc3)C)=O)C2)CCCCN1C(=O)C(N)=O 40404,C(CCCCCCC(=O)NC(CNC(=O)CC(C)C(C)C)C1CC1)SC 40405,c1(OC)ncc(C(=O)N(C2C3CN(C(c4cnc(OC)s4)=O)CC23)C)nc1C 40406,CC(O)(CCNC(N1CC2(CCC2)C1CO)=O)C(F)(F)F 40407,c1(C(N(C(C)CNC(=O)CCc2cncc(F)c2)C)=O)ccc(N)c(N)c1 40408,N1(C(CCOC(C)=O)=O)CC(C2CC2C(=O)N(C2CCOCC2C)C)C1 40409,N1(C(C(C2(O)CCCCC2)CC)=O)CCN(C(c2cnc(O)n2C)=O)CC1C 40410,C1(NC(Cn2c(C)c(Cl)cn2)=O)CC2CCC1N2C(C1(C)CC=CC1)=O 40411,CC1=C(C(=O)NC2CCC(NC(c3cn(C)nc3Cl)=O)C2)C=C2CCCN=C2N1 40412,CCCCCCOC(C)C(=O)NCC(CC)NC(c1ccnn1C1CCCC1)=O 40413,C1(C)(C(=O)NCC2CCN(C(COCC)=O)C2)CNC(=O)C1 40414,N1(C(C2(OC)CC2)=O)CCC(O)(CNC(=O)CC2CCN(C)C2=O)CC1 40415,N1(C(C2(CC=C)CCN(C(=O)C=CCN3CCC3)C2)=O)CCCCC(OC)C1 40416,C1(C2CCN(C(C3CC4CC3C4)=O)CC2)(NC(CCC(CCCC)C)=O)CCC1 40417,C(c1ccc(C2CC2C)o1)=CC(=O)OC.C1(=O)C(C)=CCO1 40418,C1(COCCO)CC=CCN1c1nnnn1CC1CC2CCCC12 40419,C1(CNC(C(CC#C)C2CC2)=O)(NC(c2nccnc2C)=O)CC2CCC1CC2 40420,C1(CCCNC(=O)CNC(c2cscn2)=O)CCCCN1C(C1CC12CCC2)=O 40421,n1(CCC)cccc1C(=O)NCC1OCCC1C(=O)NCCSCC(C)C 40422,C(C(C)C(=O)NCCNC(c1cc(C2(C)COC2)no1)=O)OCC 40423,N1(C(C=CC(=O)N(C)C)=O)CC(CO)C1(C)C.c12cc[nH]c1C(=O)NC2 40424,C1(C#N)(C(=O)NC2CC(C)(NC(CCC=CCC=C)=O)C2)CC2CC2C1 40425,Cc1[nH][nH]c(=N)c1C(=O)NCCCCCCN(C)C(c1coc(C(F)(F)F)c1)=O 40426,C1(NC(c2c(C(=O)NC3C(N(C)C)CCCC3)n[nH]c2)=O)CCC(C)(C)OC1 40427,CC1CN(C(=O)CN2CCC2)CCC1NC(=O)C(C)(C)C1(O)CCOC1 40428,C=CCCCC(C(=O)Nc1cccc(NC=O)c1)NC(=O)CCC(=O)CC 40429,n1(CC(=O)NC2C(NC(C(F)=CCC)=O)CC2)cc(Cl)c(C)n1 40430,N1(C(c2ccc(C)c(F)c2)=O)CCN(C(c2cncc(F)c2)=O)CC2(CC2)C1 40431,C(c1cnn(C)c1)=CC(=O)NC(CC=CC(=O)N(C1C(C)CCC1)C)(C)C 40432,C1(NC(CCC(C)OC)=O)CCCC12CN(C(=O)Cc1nc(C)sc1C)C2 40433,C1(C(N(C(CC)C)CCO)=O)COCCN(C(C2(C#N)CC2)=O)C1 40434,C(CCCCC(=O)NC1CC2CCC1O2)n1cc(CC(=O)O)nn1 40435,CC1=NOC(C)(C(N2CCCC(NC(c3cnn(CC(F)F)n3)=O)C2)=O)C1 40436,C#CC1(C(=O)N(CCC(N2CC(O)(C(N3CCCC3)=O)C2)=O)C)CC(=O)C1 40437,CCCC(C(=O)NCC1C2CN(C(c3cc(Br)ccn3)=O)CC12)OCC 40438,N1(C(C=C(C)C2CC2)=O)CC(C(=O)NCCn2ncnn2)C(C)(C)C1 40439,C(=O)(CCCCC#N)NC1CCCN(C(C(CC#C)O)=O)C1 40440,N1(C(C2(CC=C)CC=CC2)=O)CC2(CCC2NC(=O)CSS(C)(=O)=O)C1 40441,C1(C(N(CC=C)CC2CC2)=O)CN(C(C2CC(C)=NO2)=O)CC1C 40442,C1(CNC(CN(C2CCCC2)C)=O)CC(C)(C)CN1C(=O)CN1CCCCC1=O 40443,C1(NC(COCC=C)=O)CC(C)CN(C(c2c(C)coc2C2CC2)=O)C1 40444,C(CCCC(=O)NCC(c1ccco1)O)NC(c1cc(OC)n[nH]1)=O 40445,C(C(C)(C)CNC(c1ncn(C)n1)=O)N(C(C1(CCC=C)CC1)=O)C 40446,Cc1nc(C(C)C)ccc1C(=O)NCC1CCCC(NC(=O)CNS(N)(=O)=O)C1 40447,N1(C(COCCCC)=O)CCC(C)(C)C(NC(=O)CCOCC(F)(F)F)C1 40448,C1(NC(n2cc(C(C3CC3)C3CC3)nn2)C2CC(CSC)C2)COC2(COC2)C1 40449,C1(CNC(C2(C(C)=O)CC2)=O)CC(C)N(C(C2CCC=CO2)=O)C1 40450,Cc1ccccc1C(=O)NCC(C)CNC(=O)CCCc1cncs1 40451,C(C(CNC(=O)OC(C)(C)C)CO)NC(C1N(C(C2(OCC)CC2)=O)CC1)=O 40452,c1(N2CCN(CC(C)(F)F)CC2)nc(N2CCC(N(C)C)CC2)nc2scnc12 40453,c1(OCCCC)ccc2cc(C(=O)NC3CCN(C(=O)CC#N)C3(C)C)[nH]c2c1 40454,C1(NC(CCc2nc(=N)[nH][nH]2)=O)CCC2CCN(C(c3csc(Cl)c3)=O)C12 40455,c1(OCCC)cccnc1NC(N1CCC(CC)(CC)C1)=O 40456,N1(C(Cc2c(C)con2)=O)CCC(C)(C)C(CNC(c2cc[nH]c2C(C)C)=O)C1 40457,C1(C2CCOCC2)(C(N2CC(NC(C(C(=O)OC(C)(C)C)C3CC3)=O)C2)=O)CC1 40458,c1(C(N(C(c2ccccc2)CNC(C2CCNC2=O)=O)C)=O)cc(Cl)ncc1N 40459,C1(NC(=O)Cc2cccnc2O)C2CC3CN(C(C4CCCS4)=O)C1C3C2 40460,N1(C(c2c[nH]c(=N)s2)=O)CCC2(CNC(C3Cc4cccnc4C3)=O)CCCC12 40461,C1(CN(C)C)CCN(C(C2CC(F)CN2CC(N)=O)=O)CC1 40462,c1(C(=O)NC(CCOC)CNC(=O)CC(C)CF)ccc(S(N)(=O)=O)c(F)c1 40463,C(=O)(C1=CC2(CN(C(=O)C=Cc3ccnn3C)C2)OC1)N1C(CC)CNC(=O)C1 40464,N1(C(c2cc(C(C)=O)c(C)o2)=O)CC(NC(C2CCCSC2)=O)CC(F)(F)C1 40465,C12(C(N3CCN(C(c4ccc(C)c(C)c4)=O)C(C)C3)=O)CCCC1CC(=O)C2 40466,CC1(C)CCC(CNC(=O)C(C2CCCCC2)O)N(C(=O)CN2CCSCC2)C1 40467,c1(C(=O)NC2C(C)CN(C(c3ccoc3)=O)C2)cccc(C(N)=O)c1N 40468,N1(C(COCCCC#C)=O)CC2CCN(C(c3nnccc3C)=O)CC2C1 40469,N1(C(c2n[nH]c(C)c2O)=O)CCC(C(=O)NC(c2nncn2C)C)C12CC2 40470,C1(C(N2C(CN(C(c3scc(OC)c3)=O)C)CCC2)=O)(OC)CS(=O)(=O)C1 40471,C1(C(=O)NCC2CCC(CNC(CNC(C)=O)=O)CC2)CCCCC1(F)F 40472,c1(CN(c2snc(C(=O)OC)n2)C)cc(C#N)ccc1F.C12CCN(C1)C2=O 40473,C1(NC(CSCCC)=O)C2CCN(C(c3cnn(C(C)C)c3F)=O)CCC12 40474,CCC(C)(CCC(C)C)C(=O)NC1CCC(C(N2CCC(O)C(O)C2)=O)CC1 40475,c1(-c2cc(C)[nH]c2C)csc(=Nc2cccc(F)n2)n1CCC1CCSC1 40476,C=CCCC(C)NC(c1cc(C2CCC2)[nH]n1)c1nnnn1CCCF 40477,C=CC1CN(C(C2(c3ccc(F)cc3)CCOCC2)=O)CC1NC(=O)CCF 40478,C=CCC(C(=O)NC(CNC(c1cnc2[nH]ncc2c1)=O)C1CC1)C(C)C 40479,c1(NC2(c3nnnn3C3CC(F)(F)C3)CC(COC)C2)nc2cc(Cl)cnc2[nH]1 40480,C(=O)(C(C)(C)C1=CCN(C(=O)CC2CCCC2C)C1)NC1CC(SC)C1 40481,N1(C(C2(OC)CC(C)C2)=O)CC(C2(NC(C3COCC(C)(C)O3)=O)CC2)C1 40482,c1(OC)ncc(C(=O)NCC2(O)CCN(C(c3n[nH]cc3C)=O)C2)c(C)n1 40483,c1(NC2CCN(C(C3CC34CC(O)C4)=O)C2)ncc2ccsc2n1 40484,C12(C(=O)NCCC3CCCC3)COCC1CN(C(=O)CCc1csnn1)C2 40485,C(=O)(CC(C)CC(C)C)NCC(CCC)C(=O)N1CCC12CC(C(N)=O)C2 40486,c1(CN(C)C(C2(N(C)C)CC2)=O)ccc(CNC(C2CCCS2(=O)=O)=O)cc1 40487,c1(CNC(c2n(CC)ccc2)=O)ccc(F)c(CC(=O)OC)c1 40488,CC1CN(C(=O)C(=O)NC2C3CCCC2CC(N)C3)CCS(=O)(=O)C1 40489,Cc1cn2cc(CC(=O)NCC(C)CNC(=O)CC(C)CF)nc2s1 40490,c1(C(=O)NCC(C2CC2)NC(CCC(=O)NCC)=O)nccc(Cl)c1Cl 40491,n1(CCOCC)cc(CCCC#N)nn1.C1(=O)C(F)(F)C2(CCC2)N1C1CC1 40492,C1(NC(CCc2c(C)noc2)=O)CC=C(C(=O)N2CCC(CCO)C2)C1 40493,c1(C(=O)NC(c2ncc[nH]2)CC)ccc(CNC(=O)COc2ccsc2)s1 40494,CC1=C(C(=O)N2CCC(O)(C(C)NC(=O)C(C)NC=O)C2)COCC1 40495,Cc1ccc([N+](=O)[O-])cc1C(N1CCC(F)(F)C(NCc2cnn(C)c2C)C1)=O 40496,N1(S(C(C)C#N)(=O)=O)CCC2(COCCN2C(C2CC2(F)Cl)=O)C1 40497,C1(C(=O)NCC2CCCC(CNC(c3c(C)nsc3)=O)C2)C2CCC(F)(F)C12 40498,c1(CC)sc(C(=O)NCCC2CN(C(c3cc(CC(C)C)[nH]n3)=O)C2)cc1C 40499,C(CCCC(=O)N1CC(C(=O)NC2CC(C(F)F)C2)OC(C)C1)(OC)OC 40500,CCCCC(CC)C(=O)N1CC(C(=O)NCCN2CCC2)CC1(C)C 40501,C1(C(=O)NCC(CNC(c2ccn(CCCC)n2)=O)(C)C)C2CCC(=O)C12 40502,c1(C(=O)NCc2c(CNC(CCCC#CC)=O)cccc2)cnc2[nH]nnc2c1 40503,N1(C(C2CCC(CC)O2)=O)CCC2(NC(c3cc(C)ccc3F)=O)CCCC12 40504,c1(NC(c2cncc(CC)c2)=O)ccc(NC(c2cnc(O)cc2C)=O)c(C)c1 40505,CC1(NC(c2ccc(F)cn2)=O)CCN(C(=O)C=CBr)C1 40506,Cc1occc1C(=O)N(C)CC1(O)CN(C(=O)C(C)(O)C2CCOC2)C1 40507,C#Cc1cncc(C(=O)NCC(CNC(=O)Cc2ccc(Br)cc2)OC)c1 40508,c1(C(=O)OCC)[nH]c(C)c(C(N2CCN(CCSc3ccc(Cl)s3)CC2)=O)c1C 40509,C(=O)(C(Cc1ccco1)NC(C1CNC(=O)O1)=O)N(CCCC)CCO 40510,Cc1c(C(N2CC3CN(C(=O)CN(C)C4CC4)CCC23)=O)nc2sccn12 40511,C1(C(=O)NCC(CNC(Cc2c(C)ncnc2C)=O)C)OCC2CCCCC12 40512,CCC(CC(=O)NC1CCC(C)(NC(c2cnn(C)c(=O)c2)=O)CC1)CC(C)C 40513,c1(SCC(N2CCC(NC(C3(c4cc(C)no4)CC3)=O)C2)=O)ccc(F)c(Cl)c1 40514,CCCCC(CC)C(=O)NC1CC(C)(C(=O)N(C)Cc2ncc[nH]2)C1 40515,C(=O)(C1=CC2CCC(C1)C2)NCC(CO)NC(CCC1C(C)C1)=O 40516,c1(C(N2CC(C)NC(=O)C2)=O)ccc2c(n1)CCN(C(=O)Cc1ccccc1)C2 40517,CCCCCC(C(=O)NC1CCC(NC(=O)Cc2cn(C)nc2Cl)CC1)C(C)C 40518,c1(C(=O)NCC(CNC(COC)=O)C)oc2ccccc2c1CSC 40519,c1(CNC(C2(NC(CCC=CC(C)C)=O)CCC2)=O)ccc(F)c(F)c1 40520,C1(C(N(C2CCN(C(=O)C=C(Cl)Cl)CC2)CC)=O)C2CCC1(c1ccccc1)C2 40521,N1(C(CC2CC(OC)C2)=O)CCCC1(C)CNC(=O)CC1CCC=CCC1 40522,C1(C(N2CC(CNC(c3cncc(C)n3)=O)OCC2)=O)CCCCC1(C)C 40523,C(C(F)(F)C(N)=O)NC(C1(CCC=C)CN(C(=O)CN2CCC(C)C2)C1)=O 40524,Nc1cc2c(cc1C(=O)NC1CCC(NC(C3CC3(Cl)Cl)=O)CC1)CCC2 40525,C(=O)(CCCC(F)(F)CO)NC1(C)CCN(C(C23CCOC2CCOC3)=O)CC1 40526,C1(F)(CNC(C(SC)SC)=O)CCN(C(=O)C=Cc2cn(C)cn2)CC1 40527,c1(NC(=O)NC(C2COCCO2)CC)ccc(OC)cc1S(C)(=O)=O 40528,Cc1nc(C=CC(=O)N(C2CCC(NC(=O)Cc3ccco3)C2)C)cs1 40529,c1(SC)ccc(NC(=O)NCCOc2cccc(F)n2)cc1C#N 40530,N1(C(c2ccn(CCC)n2)=O)CCC(C)(C)C1CNC(=O)C(C)(CC)CO 40531,c1(C2(C(=O)OC)CC2)ccc(Cl)c(Cl)c1.CCC(C)(C)NC(=O)CSSC 40532,c1(C(N2CC(C(=O)Nc3ccc(O)nc3)SCC2)=O)cn2ccc(Cl)cc2n1 40533,c1(OC)cc([N+](=O)[O-])c(OC)cc1NC(C1CCN(C(c2cnc(Br)s2)=O)C1)=O 40534,C1(O)(C(=O)NC(C2CN(c3cc(CC(C)C)ncn3)C2)C)CC2CCC1C2 40535,N1(C(Cc2cnc(C)s2)=O)CCCN(C(c2cc(C)n(C)c2)=O)CC1CO 40536,C(=O)(CCCCc1ccc(Cl)cc1)NCC(CNC(Cc1cc(C)sc1)=O)O 40537,C(C)(CN1CCOCC1)(C(C)C)NC(=NC)NCc1cccc(C2OCCO2)c1 40538,C1(N(C(Cn2ncc(NCC=C)c2)=O)C)CCN(C(=O)OC(C)(C)C)CC1C 40539,Cc1cc(N2Cc3ncsc3C2)nc(=NCCCc2nnnn2C)[nH]1 40540,N1(C(c2cc(C)c(F)c(C)c2)=O)CCC2(CC(NC(=O)C(F)Br)CO2)C1 40541,c1(C2CN(C(=O)OC(C)(C)C)C2)nnc(S)n1C.N12CCC1(C)C2=O 40542,C#CCCCCC(=O)N1CCCC(C)(CNC(=O)C(CCC)OC)C1 40543,C1(C(N2C(C#C)CCCC2)=O)CN(C(=O)Cc2cnnn2C)CCC1(C)C 40544,N1(C(c2cc(OC)n(C)n2)=O)CC2CC(NC(=O)C(O)C3CCC3)CC1C2 40545,c1(CC)cc(C(=O)NCCC2COCCN2C(=O)CCC2CCC2)ccc1Cl 40546,Cc1cc(F)c(C(N2CCC(C)(CNC(=O)C=Cc3cncs3)C2)=O)c(F)c1 40547,Cc1cc(CO)cnc1C.c12ccc(cc1)C(C(=O)NC1(C)CCCCC1)N2C 40548,CC1CN(C(c2ccncc2F)=O)CC1CCNC(=O)CC1CCC(F)(F)C1 40549,CC1CC(C(=O)N(CCNC(c2ccsc2)=O)CCc2ccccc2)CC(C)C1 40550,N1(C(C(c2cnn(C)c2)C)=O)CCC(C2(NC(=O)Cc3cc(Cl)n(C)n3)CC2)C1 40551,C1(NC(C(C)OC)=O)CCC(NC(=O)Cc2cnn(C)c2C)CC1 40552,c1(CNC(c2nnnn2CCCOC)(COCC)C2CCC2)cccc(Cl)c1C 40553,N(C)(S(=O)(=O)N(C)C)CC(=O)NC(C)CNC(c1cn(C2CCCC2)nn1)=O 40554,C1(NC(C=CC=CC)=O)CCC(C)(CNC(=O)CC2(OC)CCOCC2)C1 40555,C=C(C)CC(C(=O)NCC(O)C(=O)NC(C)CCCCCO)OC 40556,C1(C#N)(CN(C)CC2(C)CC3CC3C2)CCCCC1 40557,N1(C(C(CCF)NC(C(C=C=C)C)=O)=O)CCOC(C)(C)C1 40558,c1(OC(C(=O)N(CC(CNC(C2N(C(C)=O)CSC2)=O)O)C)C)ccc(C)cc1 40559,N1(C(c2c(CC)n(CC)nc2)=O)CCCN(C(=O)CC2(OC)CC2)C(C)C1 40560,c1(C(=O)NC2C(NC(C3(COC)CCCC3)=O)C2)cc(F)c(N)c(F)c1 40561,c1(OC)cc(NC(C2CCCN2C(c2ccc(C)nc2O)=O)=O)ccc1O 40562,N1(C(c2c(CC)cccn2)=O)CCCC12CCN(C(C1CC=CCC1)=O)C2 40563,c1(CC(=O)N(CCC2N(C(C(C(C)C)OC)=O)CCCC2)C)cc(F)ccc1Cl 40564,c1(C(=O)NCC(CC)NC(=O)C(C)(C)C(N)=O)ccc([N+](=O)[O-])cc1 40565,N1(C(c2c(COC)cc[nH]2)=O)CC(CNC(=O)C=C2CCN(C)C2)CC1(C)C 40566,Cc1nc(C(=O)NC2(CNC(C3(C)CC=CCO3)=O)CC2)ccc1C#N 40567,Cc1occ(C(F)(F)F)c1C(=O)NC1CN(C(=O)C(c2ccccc2)C)CC1O 40568,CCCC(C(=O)NC)NC(=O)Cn1cc(C(C)(C)F)nn1 40569,C1(Sc2nnc(N(c3ccccc3)C)s2)CCOC(c2cccc(F)c2)C1 40570,C(=O)(C=CCNC(=O)COC(C)=O)N(CC=C)CCO 40571,N1(CC2(O)CCN(c3c(OC)cccn3)CC2)CCC2(CCCC2)C1 40572,C1(CNC2CC(OC)C(OC(=O)C3CC3)C2)CCCN(C(C)=O)CC1 40573,c1(CC(=O)NC(CC)CNC(C23CCC2C3)=O)nnn(-c2cccc(Cl)c2)c1C 40574,C1(C(N2CC3N(C(c4cc(C(CC)C)no4)=O)C(C3)C2)=O)CNC(=O)CC1(C)C 40575,N1(C(c2c(C)cns2)=O)CCOCCC1C(=O)NC1CCC(C(N)=O)C1 40576,C1(C2CCN(C(C3CCC(C)S3)=O)CC2)(NC(c2n(CCC)ccc2)=O)CCC1 40577,C(=O)(C(C)(C)CCF)N1CCCC(N2CCN(C(CC=C(C)C)=O)CC2)C1 40578,c1(C(=O)NC(C(C(C)C)C)CNC(c2cccnc2S)=O)noc2c1CCCC2 40579,CC1(C)CCC(C(N2CC=CC2(C)C(=O)NCCN2C(=O)CNC2=O)=O)C1 40580,N1(C(c2ccccn2)=O)CCC(NC(C2(Cc3ccccc3)CC2)=O)C1CO 40581,C1(NC(c2cc(CCC)on2)=O)CCCN(C(=O)C=C(C)C(C)C)C1C 40582,C1(O)(CCNC(C2CC3CC3C2)=O)CCN(C(c2ccc(O)nc2)=O)CC1 40583,c1(C(N2CC(CNC(CCC3CC(C)C3)=O)OCC2)=O)ccc(F)c(Cl)c1N 40584,Cc1c(Br)csc1C(N1CC(CC(C)NC(=O)C(C)C2CCC2)C1)=O 40585,C(C(=O)N1CC(O)C(O)CO1)C1N(C(c2ncc(CC)cn2)=O)CCC1(C)C 40586,C1(C(=O)NC2C(OC)CN(C(C3(C4CCC4)CC3)=O)C2)CCC(C)(O)CC1 40587,C1(CNC(C2CCCC(NC(CC(C)F)=O)C2)=O)CC12CCOCC2 40588,C1(C)(C(=O)NCCOCCC(N2CC(C(CC)CC)C2)=O)CCC(=O)N1 40589,C(=O)(C(C)CC(C)(C)C)N1CCC(N(C(Cn2ncc(CC)c2)=O)C)C1 40590,c1(N(CC(O)CF)C)ncc(S(=O)(=O)NCC2CC(=O)N(C(C)(C)C)C2)cc1Cl 40591,CCCCCCC(C)C(=O)N1CCCC1CN(C)C(C1CCCCN1N=O)=O 40592,N1(CC(N2CC(NC(=O)CSc3ccncc3)C2)=O)CCCCCCC1=O 40593,C(=O)(C1=CCOCC1)NC1(CO)CN(C(c2c(C(C)C)n(C)nc2)=O)C1 40594,Cc1cc(NC(=O)C(=O)NCCc2ccc(Br)s2)ncn1 40595,C(c1ccncn1)=CC(=O)NCCN(C(=O)C(C1CCOC1)SC1CC1)C1CC1 40596,Cc1cccc([N+](=O)[O-])c1C(N1CC(N(C(=O)CC2OCCC2C)C)C1)=O 40597,c1(CC(=O)NCC(C)(CO)NC(C2CCN(C)C2=O)=O)c[nH]c2cccc(Cl)c12 40598,C(=O)(CS(=O)C(F)(F)F)NC1C(CO)CCN(C(CCCNC(C)=O)=O)C1 40599,CC1CCc2ncc(C(N3CCC(NC(c4cnc(C(C)(F)F)s4)=O)C3)=O)n2C1 40600,N1(CC(=O)NC(C)CN(C(=O)C(C)C2CCC2)C)CCCNS1(=O)=O 40601,N1(C(C2CC(N(C)C)C2)=O)CCC(C)(CNC(C2CC3C=CC2C3)=O)CC1 40602,N1(C(c2oc(C)c(CO)c2)=O)CCN(C(C2(C)CCCS2)=O)CC1CC(F)(F)F 40603,N1(C(C2CN(C(C)=O)C2)=O)CC(C(=O)N(c2cc(C)cc(C)c2)C)OC(C)C1 40604,N1(C(c2c(N)nccc2)=O)CCC=C(CNC(=O)CCN2CCCC2)C1 40605,CCCCC(C)C(=O)N1CC(C(=O)N(CC)CC2CCOC2)C(F)C1 40606,c1(C(N2CC(C#N)OCC2)=O)cc(-c2cccc(OC(F)F)c2)c2[nH]ccc2c1 40607,C[S+](C)CCC(O)C(=O)N1CC(O)(CCNC(=O)COC2CCOC2)C1 40608,c1(C(=O)NCC2N(C(c3ncn(CC)n3)=O)CC(O)C2)cc(C(C)C)nc(O)c1 40609,c1(C(C(=O)NC)N(C2CCC(F)(F)CC2)C)ccc2c(c1F)CCC2 40610,c1(C(=O)NCC(CNC(C(CC)(C)OC)=O)CO)ccnc2ncccc12 40611,c1(C(N2CCC(CNC(C(C(=C)C)(C)O)=O)CC2)=O)ccc2c(C)nn(C)c2n1 40612,N1(C(c2c(CC)ncs2)=O)CC2CN(C(c3cnc(C(C)(C)C)o3)=O)CC(C1)O2 40613,c1(N2CC3OCCN(CCN(CC)CC)C3C2)cc(C)c(S(=O)(=O)NCC)cn1 40614,C12(C(=O)Nc3c(CC)cccc3C)CCN(C(=O)CC(O)C(C)C)CCC1C2 40615,Cc1ccc(CN2CCCC2CCC(=O)Nc2ccnc(OC(C)C)c2)cn1 40616,c1(C(N2CCC3CCN(C(CC=C)=O)C3C2)=O)cnc2c(c1)OCC(=O)N2 40617,N1(C(Cc2c(C)occ2)=O)C(C)C2CC1C2NC(c1cccnc1O)=O 40618,N1(C(COCC#C)=O)CCC(NC(=O)CCc2cccs2)C1C1CC1 40619,c1(OC)cc(N)ccc1C(=O)NCCN1CCC(NC(=O)C=CCO)CC1 40620,C1(C(F)(F)F)(NC(c2c(C3C(C(=O)OC)CC3O)cccc2)=O)CCC(C)(C)C1 40621,C(N=c1ccc([N+](=O)[O-])c[nH]1)C1OCCN(C(C=CSC)=O)C1 40622,c1(C(N(C)CCNC(=O)C(C)(C)COC2CCCC2)=O)cccc2nsnc12 40623,c1(OC)cc(F)c(C(=O)NC2COCC2NC(C2CN(CC(C)C)C2)=O)c(F)c1 40624,c1(C(=O)NC2CCC(NC(C(C(C)C)(C)O)=O)C2)cc(S(N)(=O)=O)ccn1 40625,N#Cc1cc(C(=O)NCC2CC2NC(c2c(Cl)ccc(F)c2F)=O)c(N)nc1O 40626,C1(NC(C2=NOC(C)(C)C2)=O)CCC2CCN(C(C3(C)CCCNC3=O)=O)C1C2 40627,c1(NC(c2cc(-c3ccc(C)o3)[nH]n2)=O)nccnc1C(=O)Nc1ccccc1 40628,CC1CCCCC1(CNC(c1ccc(O)c(O)c1)=O)NC(c1c[nH]ccc1=O)=O 40629,Cc1cccc([N+](=O)[O-])c1C(=O)NC1CC2CC(C1)N(C(=O)Cc1cccs1)C2 40630,C1(CNC(c2scc(C)c2)=O)CC(NC(c2coc(N(C)C)n2)=O)C12CCC2 40631,C(=O)(C(O)CCNC(C1COCCN1C)=O)NC(c1cc(C)no1)(C)C 40632,C1(CNC(c2c(CC)cncc2)=O)N(C(=O)CCNS(C)(=O)=O)CCCC1(C)C 40633,C(=O)(CCCNC(=O)C(C)Cn1ccnc1)N(CCC(=O)OC)CC=C 40634,c1(CC)nc(C)[nH]c1C(=O)NC1CC(CCNC(=O)Cc2[nH]cnc2C)C1 40635,CC1(CNC(C2CC2F)=O)CCCN(C(=O)Cc2c(Cl)cccc2Cl)C1 40636,c1(CC(C)NC(=O)COC2CN(C(=O)C(C)C3CCCC3)C2)ccc(Cl)s1 40637,C1(C(C)C)N(C(c2cncn2C)=O)CC12CCN(C(C1CC1F)=O)CC2 40638,N1(Cc2cn(Cc3c(Cl)nc(OC)n3C)nn2)CCCCNC(=O)C(F)(F)C1 40639,CC(C)(C)C(CC(=O)NCCC1CCN(C(=O)CN2CSCCSC2)C1)C(F)F 40640,c1(C(=O)NCC2(NC(C3CC34CC4)=O)CCC2)ccc(C2CC2(F)F)cc1 40641,CN1CCOCC1C(=O)NCC1(C(N2CC=CC2CF)=O)CC1 40642,Cc1c(C(=O)NC(C)CNC(=O)CCc2ccon2)ccn1C 40643,c1(C(N2CC=CC(C(N3C(COC)CCC3)=O)C2)=O)cc(S(=O)(=O)NC)cn1C 40644,C(=O)(C1=NOC2(CCN(C(C3(CN)CC3)=O)C2)C1)Nc1cnc(C)c(Cl)c1Cl 40645,N1(C(COCCOC)=O)CCC2(CCCCN(C(c3coc(COC)n3)=O)C2)C1 40646,C12(CNC(C(C3CC3)OC)=O)CCCC(CN(C(=O)C(C)(C)c3ccno3)C1)C2 40647,Cc1cc(OCCC(N2CC(C)C2c2ccccc2)=O)no1 40648,c1(N2CC(NC(C3C(C)(Br)C3)=O)(CO)C2)ncncc1Br 40649,N1(C(C2C(C)(C)CC2)=O)CCCCC1C1CCN(C(c2cc(Br)no2)=O)CC1 40650,N1(C(c2c(CC)n(CC(C)C)nc2)=O)CCCC(CNC(C2CC(=O)N2)=O)CC1 40651,N1(C(C(C2CCN(C(=O)C(N3CCOCC3)C)C2)C)=O)CCC(O)C(C)C1 40652,C1(C(N2CCC(C(=O)OC)C2(C)C)=O)CC2C=CC1N(C(=O)C(C)n1ccnn1)C2 40653,Cc1sc(C)c(C(N2CC3(CC(NC(=O)C(C)CC(N)=O)CO3)C2)=O)c1C#N 40654,C1(C(N2CC(F)(C(N(C3CN(C4CC4)C3)C)=O)C2)=O)CC2CCC2C1 40655,CC(c1ccccc1)=CC(=O)NCC1CCC1NC(C1(CCN(C)C)CC1)=O 40656,N1(C(C(C)CC(F)(F)F)=O)CCCC2(NC(=O)CN3CCC3)CCCC12 40657,C1(CC(=O)NCC(C(C)C)(C)C)C2CCC(C2)N1C(=O)CCCn1cncn1 40658,c1(C(N2CCCC(CN(C(c3n(CC)ccc3)=O)C)C2)=O)c(OC)ccnc1F 40659,N1(C(COCC#C)=O)CCN(C)CC1CNC(=O)CSc1n[nH]c(C)n1 40660,c1(C(N(CCC(=O)N(C)Cc2cn(CC)nc2)C(C)C)=O)ccc(O)nn1 40661,N1(C(C=C(C)Cl)=O)CCC2(NC(=O)COc3cccc(C)c3)CCCC12 40662,Cc1ccsc1C(=O)N(CCC(=O)NC(C)(C)CO)C 40663,C(=O)(CCCS(=O)(=O)N1CCCC1)NC(CN(C(COCCC#C)=O)C)C 40664,c1(OC)cccc(Cl)c1CC(=O)NC1CCN(C(=O)CC2OCCO2)C(C)C1 40665,c1(COCC(=O)NCC(CN(C(CN(C)CC)=O)C)C)ccnc(O)c1 40666,N1(C(CC(C)C)=O)CC2CCCC1CN(C(=O)Cc1ccc3nc(O)[nH]c3c1)C2 40667,C(=O)(CCCC(C)(C)C)NCc1cn(CC(=O)NC(CC(C)C)C(N)=O)nn1 40668,N1(C(C(C)S(N)(=O)=O)=O)CCC2(CCCC2NC(c2cc(Cl)cn2C)=O)CC1 40669,C(CCCC(=O)NCC1(O)CN(C(c2cn(C(C)C(F)F)nc2C)=O)C1)NC(C)=O 40670,N1(C(c2ncc(NC)nc2)=O)CCC(C(=O)N(C)CC2CCN(C)C2)=C(F)C1 40671,O=C(C1=CC2CCCC12)NCC1CC(F)(CNC(c2ncnc(O)c2Br)=O)C1 40672,CCC(C)C(O)C(=O)NCC(CO)NC(c1ccc(F)c(C(F)(F)F)c1)=O 40673,CCC(C(=O)OC)C(=O)OC(C)(C)C.C1(C2CCCCCC2)CCCC2(CC2)NC1=O 40674,C#CC1(C(=O)NCCN2CCOC(C)C2)CCN(C(=O)CC2CSC2)CC1 40675,c1(C(=O)NCC2CC(NC(c3c(OC)nn(C)c3)=O)C2)ccc(F)c(Cl)c1 40676,c1(C(N2CC(CNC(c3ccco3)=O)C(C(F)(F)F)C2)=O)cnc(F)c(F)c1 40677,Cc1[nH][nH]c(=N)c1C(=O)NCCCN(C(c1coc(Cl)n1)=O)CC1CCCC1 40678,C1(CNC(=O)CNC(c2cccs2)=O)CCN(C(C2(CCO)CC2)=O)CC1(F)F 40679,c1(NCC#CC)ncnc2c1ncn2C(CC(=O)N(C)C)C1CC1 40680,c1(C(N(C2CCCN(C(CC(C)F)=O)C2)C)=O)ccc2oc(S)nc2c1 40681,C1(C(=O)NCCN(C)CC)CCCN(C(=O)CC2(OC)CCC2)C1C 40682,C1(CC(=O)NCC2CCC(C(=O)NC(CC(C)SC)=O)C2)CCCC2CC12 40683,N1(S(CCC)(=O)=O)CCC2(CCOCC2)C(c2cnn(CCC)c2)C1 40684,N1(C(CC=C=C)=O)CCC(NC(c2ccn(-c3ccccc3)n2)=O)C1C(C)C 40685,c12cc(ccc1F)NC2=O.c1(C(C)C)cc(NC(C2CN(C(N)=O)C2)=O)on1 40686,c1(CC)cc(C(=O)NCC(C)CN(C)C(C2(COC(C)C)CC2)=O)oc1CC 40687,c1(C(=O)NCC(CC)NC(c2cnn(CCO)c2C)=O)cccc(F)c1OC 40688,C(=O)(C1=CC2CCC=CCCC12)N1CC(C(C)NC(c2cn(C)c(=O)n2C)=O)C1 40689,C1(NC(=O)CS(=O)(=O)NC2CC2)CN(C(=O)C=CBr)CC2(CCC2)C1 40690,N1(C(c2cc(CNC(c3c(C)ocn3)=O)nn2C)=O)CC2(CC2)CC1CO 40691,C=C(F)C1(CC(=O)N(CCC(=O)NCCc2ncn(C)n2)CCCO)CCC1 40692,c1(NC(N(CC(C(C)C)OC)C)=O)c2c(c(Br)c3c1CCC3)CCC2 40693,O=C(N=c1[nH]ccc2cc(Br)ccc12)C1CC1N.c1c(Cl)cc(F)cc1Cl 40694,C(=O)(C1=C(C)CCOC1)NCC(CNC(C1(C)COCCO1)=O)OC 40695,C1(C(=O)NCC2C(=O)CC2)CCCN1NC(=O)c1cn2c(n1)CCC2 40696,N1(C(c2ccc(OC)o2)=O)CCN(C(=O)CC(=O)N(C)C)C2CCCCC2C1 40697,c1(C(N2CCCC(N(C(C3CC=C(C)CC3)=O)CCF)C2)=O)cc2n(n1)CCC2 40698,c1(OCc2cn(CC(CNC(c3ccc(CC)o3)=O)OC)nn2)cccc(F)c1 40699,C12(CCCOC(CCCC#C)=O)CCC(C1)N(C(C1CCC(=O)N1C(C)=O)=O)C2 40700,C1(OC)CN(C(=O)CCN(CC(F)(F)F)C)CC1NC(=O)Cc1cccn1C 40701,Cc1ncnc(C)c1CC(=O)NCC(CNC(=O)CCC1OCCO1)C(F)(F)F 40702,CC1CCN(C(C2CC(=O)NC(=O)C2)=O)CCN1C(=O)C=CC=C(Cl)Cl 40703,C1(C)(CC)CCN(C(C2(CNC(=O)C(C)O)CCC2)=O)CC1 40704,C1(C(N2C(CCNC(=O)Cc3ncc(Cl)s3)COCC2)=O)CC2CCC(C1)C2 40705,C1(CNC(c2c(C)ncs2)=O)CN(C(c2ccc(F)cn2)=O)CC1C(F)(F)F 40706,Cc1nnc(NCC(C)N(C)C(c2ncccc2Cl)=O)c(C#N)c1C 40707,C#CC1CC2(CC2)CN1C(C1CCN(C(C2CCCCC2OC)=O)CC1(C)C)=O 40708,c1(CC(=O)NCCC(=C)CNC(=O)CCCc2ccsc2)nn(C)cc1Br 40709,C(=O)(C(CC1CCC1)NC(=O)COC1CC=CC1)NCC(C)SC 40710,c1(OC)cccc2c1OCCC2NC(c1c(Br)ccc(C(F)(F)F)c1F)=O 40711,N1(C(c2c(C)cno2)=O)CCC(O)C(NC(=O)CCOCCN(C)C)C1 40712,N1(C(c2nc(OC)oc2)=O)CC2=C(C1)CN(C(=O)CC1COCC3(CCC3)O1)C2 40713,C(=O)(C1=NNC(C(F)(F)F)C1)NC(C1(O)CCN(C(=O)CC2CCC3CC23)C1)C 40714,C1(N(C(=O)CCCc2ccsc2)CC)CCN(C(=O)C=Cc2nnn(C)n2)CC1 40715,c1(C(=O)NCC2N(C(C(C)S(N)(=O)=O)=O)CC3(CC3)C2)coc2ccc(O)cc12 40716,N1(C(C=CC=CC)=O)CCCC(N(C(c2ccccc2Cl)=O)CCO)C1 40717,N1(C(C(C)Sc2cn(CC(C)(C)O)nn2)=O)CC(C)CCC(C)C1 40718,CN1CC2(CCN(C(c3ccc(=N)[nH]c3)=O)CC2)c2ccccc21 40719,N1(C(C2C(C(=O)OC)C=C2)=O)C(C(=O)NCc2cnn(C)c2OC)CC2CC12 40720,c1(OCC(=O)Nc2c(C(=O)OCC)cncn2)cc(C)ccc1C(C)C 40721,c1(NC2(CCNC(C3(C)CC(C)OCC3)=O)CCC2)ncc2c(ncn2C)n1 40722,C1(CC(=O)NC)SC(=Nc2ccccc2)N(CC(CC)(CC)c2ccccc2)C1=O 40723,N1(C(c2cn(C(C)C)nc2)=O)CCC(C)(CNC(c2[nH]nnc2C2CC2)=O)CC1 40724,CC1(OCC(=O)NC2COCC2NC(=O)CC2SCC2)CCOCC1.C(C(F)(F)F)O 40725,c1(C(N(CCCCCCNC(C(C)=C(C)C)=O)C)=O)cc(=O)n(C)cc1Br 40726,CCC(CC(=O)N(C(C)C(=O)NC1(CCO)CCCCC1)CC)OC 40727,C1(C(N2CCC(C)(CCNC(C(CC)CC)=O)C2)=O)CCc2nc[nH]c2C1 40728,C1(CC(=O)NCC(CNC(CCOCC#C)=O)(C)C)CCC(=O)N1CC 40729,C(C)(C)(C(=O)N1CCCCO1)C1CCN(C(c2ccn(CCC)n2)=O)C1 40730,Cc1ccsc1C(N1CCC(NC(C2(CC3CC3)CCCO2)=O)C1)=O 40731,C=CCC(C)(C)CCN=c1cccc(S(=O)(=O)N2CC(C)c3ccccc32)[nH]1 40732,c1(CCCC)nc(C)c(CC(=O)NCC2(C(N)=O)CN(C(c3ncc[nH]3)=O)C2)s1 40733,N1(C(C2C3COCC23)=O)CCC2(CCCN2C(=O)C2=CCCC2)C1 40734,c1(-c2[nH]c(=NCc3c(OC)c(F)ccc3)sc2)cc(F)c(C#N)cc1F 40735,N1(CCCc2cccc(C)c2)CC2CCC1CN2C(c1nnn(C(C)(C)C)n1)=O 40736,C1(C(N2C(CCNC(C(C)(Cl)Cl)=O)CCCC2)=O)CCC2CCC1O2 40737,CCC(O)C(C)(C)C(=O)N1CC2CCCC2(NC(c2ccoc2C2CC2)=O)C1 40738,C(=O)(CCC(F)(F)Cn1cc(CCO)nn1)N1CCCC(COC)(OC)C1 40739,N1(C(c2c(OC)cncc2)=O)CCC(C)(C)C1C(=O)NCCCSCCO 40740,c1(OC)cc(Cl)c(CN2CCCN(c3nc(C4CC4)ns3)CC2)cc1OC 40741,c1(NC(c2n(CCOCC)nnn2)CCOc2ccccc2)ccc(Cl)cc1 40742,C1(N(C(c2ncn(CCNC(C(C3CC3)OC)=O)c2)=O)C)CCC(C)(C)C1 40743,C(=O)(C=C1SCC(=O)N1C)N1C2CC(NC(C(COC)(F)F)=O)CC1CC2 40744,CCC(C)(C)C(=O)NC(c1nc(C(=O)N(C)CCC2CCCO2)co1)C 40745,c1(NC(C)=O)ccc(CC(=O)N(C2C3CN(C(=O)C(F)=C(C)C)CC23)C)cc1 40746,C1(CNC(CC2CCN(C)C2)=O)CC12CCN(C(=O)Cn1nnc(=O)[nH]1)CC2 40747,Cn1nnc(CNC(=O)Cc2csc(-c3ccco3)n2)n1 40748,C1(C(=O)NCC2CN(C(CC(=C)C)=O)CC2C(F)(F)F)Cc2nccn2C1 40749,n1(CC)c(C(=O)NCCC(F)Cn2cc(C3(C)CCCC3O)nn2)cnc1O 40750,c1(C(N2CC(CNC(CC(CC)C)=O)C3(C2)CC3)=O)cnc2c(c1)nnn2C 40751,N1(C(C(CC=C)CNC(=O)CNC(C)=O)=O)CC(C)CCCC1C 40752,c1(C(=O)NCC2N(Cc3ccc(OC)nc3Br)CCC2)cccc2cn(C)nc12 40753,C1(CC=C)(NC(=O)C(c2ccccc2)F)CCN(C(=O)C(C)(C)COC(C)C)C1 40754,S(=O)(=O)(c1ccc(=NCc2cnn(C(C)(C)C)c2)[nH]c1)N(C1C(C)CCCC1)C 40755,c1(C(N2CCC(CNC(CCCSC)=O)C2)=O)ccc(Cc2ccsc2)cc1 40756,CC1(C(=O)OCC2CCOCO2)CN(C2CCCCC2)C1 40757,C(C1CCCN1C(c1cc(C)sc1N)=O)=CC(=O)NC1(CC)CCOC1 40758,c1(OC)ccc(F)cc1CC(=O)NC1C2CC1N(C(c1cc(C(C)C)on1)=O)C2 40759,C#Cc1cncc(C(=O)NC2CCCCC2CNC(=O)C(F)C(C)(F)F)c1 40760,C1(C(N2C(COC)CCCC2)=O)CN(C(=O)C(C)c2cc[nH]n2)CC1(C)C 40761,c1(C(N(CCN(C(C2COCC(C)O2)=O)CC)CC)=O)cc(C)c(F)cn1 40762,CN1CC(F)CC1C(=O)NC12CC1CN(C(c1cccc(CCO)c1)=O)C2 40763,N1(C(CC(CC)C)=O)CCCCCC(NC(C2OCCC2(C)C)=O)C1 40764,c1(C(=O)NC2CCN(C(c3c(C)nn[nH]3)=O)CC2C)cc2c(s1)CCSC2 40765,Cc1cc(F)c(Cl)cc1C(=O)NCC(F)CNC(=O)CC(O)C(C)C 40766,C1(NC(COC(CC)CC)=O)C2CCC1CN(C(c1cc(O)n(C)n1)=O)C2 40767,C(=O)(CC1=CCCCC1)NCC1CCCN(C(CCCOC(CCC)=O)=O)C1 40768,c1(C(C(=O)NCCCCNC(c2n(COC)ncc2)=O)C)ccc(Cl)c(Cl)c1 40769,CCC(C(=O)NCCC1(O)CN(C(C2(F)CC2(Cl)Cl)=O)C1)OC1CCCC1 40770,C1(CC(=O)N(C2CCCC2)CCNC(=O)C=Cc2cscn2)CCC(F)(F)CO1 40771,c1(C(C)C)cc(C(=O)N(C(C)C(=O)N(CC(O)CO)CCO)C2CC2)n[nH]1 40772,C=CCC(CC(=O)N1CCCC(N(C)C)CC1)NC(c1ccc(C)c(C)c1)=O 40773,C(CCN(C)C(C1CCC(O)CN1C)=O)(C(C)(C)C)NC(C(CSC)OC)=O 40774,c1(C(=O)NC(C(=O)NCC(C)N(C(COC)=O)C)C)cnc(C(C)(C)C)o1 40775,CC(C)CC(C)(C)C(=O)NCCC(C)NC(=O)COC1CCC(C)CC1 40776,Cc1nn(C)c(C)c1CNC(=O)C(C(C)O)NC(=O)OC(C)(C)C 40777,C(=O)(C1=CCCS1)NC(C1CCN(C(c2cscc2C(N)=O)=O)C1)C 40778,c1(CCNS(CC2(C)COC(=O)N2)(=O)=O)cccc(Cl)c1Cl 40779,C(C)(C)(C(C)NC(=O)C(C)=C1CC1)NC(C1(CC)CCC1)=O 40780,C(=O)(C(C)C(O)C(C)C)N1CCC(C(C)NC(C(Br)=C(C)C)=O)CC1 40781,C1(CC(=O)NCC(C)N(C)C(c2csc(C3CCCCC3)n2)=O)CC=CCC1 40782,C1(C)(CC(=O)N(CCN(C)C)CCO)CCN(C(C2(O)CCCC2)=O)C1 40783,c1(C(=O)NC(CCN(C(C(CCC)CCC)=O)C)C)ccc(=O)n2c1COCC2 40784,c1(C(=O)NCC2CCN(C(=O)Cc3ccnc(Br)c3)C2)cc2n(n1)CCO2 40785,CCC(CCC(=O)NC(C)CC(=O)NCC)OC(C)C.C1(=O)CCCO1 40786,C(=O)(C(C)(F)C(C)(C)F)NCCCC1(NC(CCc2cccc(OC)c2)=O)CC1 40787,C1(C(=O)NC(C)(C)CC2CCC2)CC2CCC1N2C(=O)CCCn1cccn1 40788,c1(CN(CCOCC)C)cc2c(cc1O)CCCC2 40789,C1(Cn2cccn2)C(=O)N(C)CCC(=O)N1.C(CC(=O)C1CC1)OCC#C.OC 40790,N1(C(Cc2ccc(CC)cc2)=O)CCC(C(C)C)CC1CNC(=O)C(C)SC 40791,C1(NC(=O)CSc2cccc(F)c2)CC(O)CN(C(c2ccc[n+]([O-])c2)=O)C1 40792,C1(NC(C(CNC(Cc2cn(SCC)nn2)=O)OC)=O)C2CCCC1CC2 40793,CC1=C(C(=O)NC2CCC2NC(c2cnn3ncccc23)=O)CCC(C)(C)C1 40794,c1(CC(=O)N(C2CCN(C(C3(C)CCCC3C)=O)C2)CC)ccccc1O 40795,C1(NC(c2ccc(OC)nc2C)=O)CCN(C(=O)CC(C)N(C)C)CC1(C)C 40796,C=CC(C)(CCOC)C(=O)N1CC(CC(=O)NC2CCC(C)NC2=O)(OC)C1 40797,C1(N(C(C)=O)Cc2c(C(=O)OC)occ2)COc2cc(Cl)ccc2O1 40798,CC1(C(=O)OCCNC(=O)COc2nc(O)nc(O)n2)CC2(CCC2)C1 40799,C1(C(=O)NCCN(C)C(c2cnns2)=O)C2Cc3c(Br)cccc3C12 40800,c1(N2C(CC)CC(C(=O)O)CC2)nc2ccc(C(F)(F)F)cc2s1 40801,C1(C(=O)NC2CC(C)(NC(C3CC(CN(C)C)C3)=O)C2)CC2(C1)CC(F)(F)C2 40802,c1(C(N2CCC(N(C(C(C(C)C)F)=O)C)C2)=O)cccn2nccc12 40803,c1(CC#N)ccc(NC(C2COCCN2S(=O)(=O)Cc2ccc(F)cc2)=O)cc1 40804,c1(CC(N2CCC(=CCNC(C3CC4CC4C3)=O)CC2)=O)cccc2c1CCC2 40805,N1(C(C2C(NC(=O)COc3ccc(F)cc3)CCC2)=O)CCN2CCC1CC2 40806,C(=O)(C(C)(O)C(C)C)NCC#CCNC(c1c(C)[nH]nc1C(F)(F)F)=O 40807,N1(C(C(CCC#C)NC(=O)Cc2ccn(CC)n2)=O)Cc2cncnc2C1 40808,C1(C(N2CC(CNC(C(C)N(C)Cc3ccccc3)=O)C2)=O)CCS1(=O)=O 40809,C12(C(N(CC)CC)=O)CC1CN(C(C1CCCN(C(c3ccc(Cl)s3)=O)C1)=O)C2 40810,C1(C2CCCCC2)(C(=O)NCC2(C)N(C(C(C)CC3CC3)=O)CCC2)CC1 40811,C1(NC(c2cc(C)c(C)nc2)=O)CN(C(=O)CCC2CCCCC2)CC1N=[N+]=[N-] 40812,C12(CC)CCN(CC1)C(=O)c1cc(n[nH]1)C(=O)N2.c1(CC23CC2C3)ccccc1 40813,c1(CNC(N2C(CC(=O)OC)C(C)CCC2)=O)ccc2c(c1)cc(C)n2C 40814,Cc1ncc(C(=O)NC(C(=O)N(CCC#N)C)c2ncco2)s1 40815,C1(C(N2CC=CC(NC(C3CCC(C)(CC)O3)=O)C2)=O)CCC(F)(F)C1O 40816,c1(CN2C(C(=O)Nc3cnccc3C(N)=O)CC(C)C2)ccc(Br)cc1Cl 40817,CC#CCCC(=O)N1CCC(N2CCN(C(c3csc(CC)n3)=O)CC2)CC1 40818,N1(C(C(C)C2(O)CCC2)=O)CCC2CCC(C1)N2C(c1cc(Br)cs1)=O 40819,c1(C(=O)NCC23N(C(CC45CC(C)(OC4)C5)=O)CC(C2)C3)cc(O)cc(=O)o1 40820,c1(-n2cc(C(C)NC(c3cc(Br)c(Br)[nH]3)=O)nn2)cccc(OCC#N)c1 40821,C1(C)(C(=O)NCC(CC=C)NC(=O)COc2cc(C)on2)CCCCNC1=O 40822,C(C)(N=c1[nH]c(=NCCCSC(C)(C)C)[nH]c2c1CCC2)c1c(C)noc1C 40823,N1(C(c2cnn(C3CC3C(=O)OC)c2)C(=O)NCCCSC)CC2CCC1C(O)C2 40824,CC(CC(F)(F)F)C(=O)NCCCN1CCN(C(=O)C(C)(C)N(C)C)CC1 40825,c1(C(N(CCNC(CCN(C(C)=O)C)=O)C2CC2)=O)c(Br)ccc2n[nH]cc12 40826,C(=O)(CC(C)OC)NCCCOCCCNC(C1C(COC)(CO)C1)=O 40827,C1(C(=O)NC2CC(CC(=O)NCc3c(C)noc3C)C2)CC(C(C)C)=NO1 40828,O=C(C1=C2CCCN=C2NN1)N1CCCC(c2cn(-c3c(Cl)cccc3Cl)nn2)C1 40829,C1(NC(c2cc(C)sn2)=O)CCC2(CC1)CCN(C(=O)CCc1cnn[nH]1)CC2 40830,C(=O)(CCC(=O)NC1CCC(CNC(c2ccn(C(C)C)n2)=O)C1)NC 40831,C1(COC)(NC(C2CC(n3cc(C4(C)CSC4)nn3)C2)=O)CCCC1 40832,c1(NC)snc(C)c1C(N1CC(CNC(c2c[nH]c(C(N)=O)c2)=O)C(O)C1)=O 40833,C1(NC(Cc2cccc(C(C)C)c2)=O)CN(C(=O)C(C)n2cncn2)CC1(C)C 40834,CC1CN(C(=O)CC(C)C(F)(F)F)CCCN1C(c1cncc(C(F)(F)F)c1)=O 40835,c1(C(C(=O)NCC=C)N(C)CCc2cccs2)cc2n(n1)CC(C)(C)CO2 40836,C1(C(c2n(C3CC(F)(F)C3)nnn2)NCCF)C(F)(F)C12CC2 40837,C1(CN=c2nc(CC)[nH]s2)CC(C)(C)CCC1NC(c1cc(C(C)C)nn1C)=O 40838,C1(N(C(CCCCOC)=O)C)CCC2CN(C(=O)Cn3nccc3C)CC12 40839,c1(C(=O)NCCC(C)NC(c2cc(C)nnc2O)=O)c2c(nn1C)CCC2 40840,C=C(F)C1(CC(=O)NCC2(C(=O)NCC3=NOC(C)C3)CC2)CCC1 40841,CC1(C)COCC(NC(=O)C(C2(C)CC2)NC(=O)Cc2cnns2)C1 40842,C1(OC)(CO)CCN(C(=O)C(CO)NC(C2SCCS2)=O)CC1 40843,c1(C(c2n(CC)nnn2)NC2CN(c3nncs3)C2)cc(C)nnc1C 40844,C1(NC(c2c(F)ncc(OC)c2)=O)CC2CN(C(C3CC=CCC3)=O)CC2C1 40845,N1(C(C(CC=CCC)C)=O)CC2CC(NC(=O)C3=C(C)CCC3)C1C2 40846,C1(C(=O)NCC(=O)N(CC(N2CCN(C(C)=O)CC2)=O)CC)CCC2CC2CC1 40847,C(C(C)C(=O)NCC1CCC(C(=O)NCc2cnn(CCF)c2)C1)SC 40848,C#Cc1cn(C)nc1C(=O)NCC1CC(NC(=O)C2=COCCO2)CC1O 40849,Cc1nc(CN=C(NC(C)C2CC2)NC2CCCN(S(C)(=O)=O)C2)c(C)o1 40850,CC(C)C(CCN(C(=O)CC1(CO)CCCCC1)C)NC(=O)CC1CCOC1C 40851,N1(C(C(CCC)OCC)=O)CC(CNC(c2cn(C)nc2O)=O)OC2(CCC2)C1 40852,CC(C)(C)C1=CCN(C(=O)COC2CCN(C(c3ccc(C(N)=O)[nH]3)=O)C2)CC1 40853,c1(C(N(C2CCN(C(C3CNC(=O)C3)=O)CC2)CCC)=O)n[nH]c(C2CC2)c1Cl 40854,N1(C(C(C(C)C)O)=O)CCN(C(=O)CCCCCC#N)CC(CO)C1 40855,C1(NC(C(CNC(C2(COC)CC(=O)C2)=O)C)=O)C(O)C2CCOC12 40856,C(=O)(C1=C(C#N)CCC1)N1C(CN(C(C(F)=C(C)C)=O)C)CCC1 40857,c1(OC)ccc(C(N2CCC(N(C)C(c3cc(F)ccc3N)=O)C2)=O)c(F)c1Cl 40858,c1(CC)c(C(=O)NC(C)C=CC(=O)NCC(C)OCCO)ccn1C 40859,C1(CN(C(CNC(C(CC)C)=O)=O)C)CCN(C(c2cc(F)c[nH]2)=O)CC1 40860,c1(CCNC(C=C(C)CNC(=O)C(C)CN(C)C)=O)ccc(C)s1 40861,N1(C(C2CCN(C(C)=O)C2)=O)CCCC2(NC(C3COCCN3C)=O)CCCC12 40862,c1(C(=O)OC)cc(F)c(F)cc1NC(C1CC(F)CN1C(c1cc(Br)c[nH]1)=O)=O 40863,C(C)(C)(CN=c1nc(NC(CCO)C(F)F)c2c([nH]1)c(C)nn2C)OC 40864,CC(CN1C(=O)CCNC1=O)C(=O)NNC(=O)C1(C)CN(C(C)(C)C)C1 40865,c1(CCCC(=O)NCC(C)N(C(=O)C(C)c2cncs2)C)ccc(C#N)cc1 40866,C(=O)(CCCC(F)(F)F)N1C(C)CC(NC(C2CCOC(=O)CC2)=O)CC1 40867,N1(C(c2cc(N)c(Cl)cc2)=O)C2CCC1CN(C(c1cn(C3CCC3)nn1)=O)C2 40868,n1(CCC(=O)NCC(C)NC(C2CCCCO2)=O)c(=O)oc2ccccc12 40869,N1(C(C2=C(C)OCC2)=O)CC2CN(C(=O)CCc3ncc(C)[nH]3)CC2(C)C1 40870,c1(CC)ncc(C(=O)NC2(CCCNC(c3ccc(CC)s3)=O)CC2)[nH]1 40871,c1(C(=O)NC(C2(O)CN(C(C3CC34CCC4)=O)C2)C)ccc(Cl)c2c1OCCO2 40872,c1(C(=O)NCCN(C(C2CN(C)C(=O)N2)=O)C)cccc(C#CCO)c1 40873,N1(C(C(C)n2ccnc2)=O)CCSCC1CCNC(C1NC(=O)CC1C)=O 40874,CC1CC(NC(C2CCC3CC3CC2)=O)CCN1C(=O)C1=CCCC1 40875,C1(CNC(=O)C=CC2CC2)CC2COCC2N1C(=O)Cn1ccc([N+](=O)[O-])n1 40876,N1(C(c2csc(Br)c2)C(=O)NCC)CCC(C2(C)CC2)CC1 40877,CCCCCCC(C)(c1nnnn1CCC)NC1CCN(C(C)=O)C1 40878,C(CN(C(=O)CC1CSCCS1)C)(CO)(CO)NC(COCCC)=O 40879,c1(C(N2CCC(NC(C(C)OC)=O)C(F)C2)=O)noc2c1COCC2 40880,C#Cc1cccc(CC(N2CCC3(NC(c4nn(C)cc4C)=O)CC3C2)=O)c1 40881,C1(C)(C(=O)NC(C2CN(C(c3cc(O)ncn3)=O)CCO2)C)COC(=O)N1 40882,C1(NC(c2occ(C)c2C)=O)CCC(C)N(C(=O)Cc2ccc(F)cc2Cl)C1 40883,C=C(C)C1CCC(C)=CC1CC(=O)NCCCCN(C(=O)CCCC(=O)OC)C 40884,N1(CC)CCOCC1C(=O)NCC1CCCN(C(=O)Cn2nnc(=N)[nH]2)C1 40885,c1(C(C)=O)cc(CC(=O)NC2CCC2N(C)C)no1.C12CC(C)(C1)C(=O)N2 40886,n1(C(C)C(=O)N(C)Cc2cncs2)cc(C2CC2CO)nn1 40887,C1(C(=O)NCC2(CC)CCC(=O)N2)CCCCCCN1C(C1CC=CC1)=O 40888,C1(NC(c2cnc(C)nc2O)=O)COC2(C1)CN(C(=O)CCC(C)CN(C)C)C2 40889,c1(C(C)COC(=O)CNC(=O)Cc2cccs2)ccncc1Br 40890,C(=O)(C1=NNC(C(F)(F)F)C1)NC(C1CN(C(=O)C(C)(C)O)C1)C 40891,c1(C(N(C(C)CN(C)C(c2csc(Cl)c2)=O)C)=O)ccc(F)c(Br)c1 40892,N1(C(CCCCC)=O)CCC(NC(c2cccnc2O)=O)C(CO)C1 40893,C(CNC(C1(C(C)(F)F)CC1)=O)(C(C)C)NC(CC1CN(C(=O)OC)C1)=O 40894,N1(C(c2cccc(C)n2)C(=O)NCC2CCOC2)C2CCC1CN(C)C2 40895,C1(NC2(c3cn(CCCC)nn3)CCC2)CCc2ncc(C)n2C1 40896,CN1CCC(C)(C(=O)NCCN(C(=O)COC2CC(F)(F)C2)C2CC2)C1 40897,C(C(CN=c1cc(NC(c2ccc(Br)cc2)CF)nc[nH]1)OC)OC 40898,C1(C(=O)NCC(c2cc(OC)c(Cl)cc2)F)CC2COCC(C1)C2(F)F 40899,C1(CNC(Cc2ccn(C(C)C)n2)=O)CC(C)(C)CN1C(C1CC(C)C1)=O 40900,C1(NC(c2ccc(C)s2)=O)CN(C(=O)CC2CC=CCN2C)CC1C 40901,N1(C(C(c2cn(C)nc2)=O)=O)CCCC(CC(=O)NCC(=O)NC2CCC2)CC1 40902,Cc1cc(C(=O)NC2CCCC(NC(=O)C3=NOCC3)C2)cc2c1NCCC2 40903,c1(-c2c(CN3CCCC(N(C)C)C3)ccnc2)cc(S(N)(=O)=O)ccc1O 40904,c1(C(=O)NC2C(N(C)C(C3CC3(Cl)Cl)=O)CCCC2)n[nH]c2c1CCOC2 40905,c1(NC(=O)NC2CC(CCNC(=O)OC)C2)ccnnc1O 40906,CC1CCOC(Cc2cn(C3CCCC3NC(=O)Cc3nccnc3N)nn2)C1 40907,CCC(C(=O)NC(C1CCN(Cc2nc(C3CC3)nn2C)CC1)C)C(C)C 40908,N1(C(N2CCN(C(COC)C)CC2)=O)CCCc2cc(C)cc(F)c21 40909,c1(CC(=O)NCCCN(C(CCC2CCN(C)C2)=O)C2CC2)cccc(Cl)c1 40910,C1(OC)(NCCC(=O)NCCC(=O)OC)CCC(C)(C)C1 40911,C(=O)(CCCC(=O)N(CCF)CCNC(=O)COCCOCCO)OC 40912,c1(C(=O)OC)nn(C)nc1C(=O)N(C)CC1CCN(C(=O)CN2CCOCC2)C1 40913,C(=O)(C1=NN(CC)C(=O)CC1)N(C)CC1N(C(c2nc(CC)oc2)=O)CCCC1 40914,c1(C)ccccc1C.c1(C(c2n(CCCSC)nnn2)NCC2CC2)nc(C)c(C)o1 40915,C1(NC(c2cccc(CNC(CC3CC(SC)C3)=O)n2)=O)CCC12CCCC2 40916,N1(C(CS(C)(=O)=O)=O)CCCC(O)(CNC(C2OCCC2c2ccccc2)=O)C1 40917,c1(NC(N2CC(C(C#C)C)C2)=O)cc(C(=O)OCC)cc([N+](=O)[O-])c1 40918,Cc1ccc(C)c(C(=O)NCC2C(C)CCN2C(=O)CNc2ccccn2)c1C 40919,N1(C(c2cnn(C)c2C#N)=O)CCC2(CC1)CC(NC(=O)C(F)C1CCCC1)C2 40920,C1(C(=O)NCC2CCCN(C(=O)CCC3CCCC3)C2)(NC(N)=O)CCCCC1 40921,C(=O)(C1=CCCSC1)NCC(c1ccc(C)cc1)NC(c1cc(=O)c(C)c[nH]1)=O 40922,Cc1ccc2cc(C(N3CCC(C(C)NC(C4CCCC4F)=O)CC3)=O)cn2c1 40923,c1(C(N2CCN(C)CC2CNC(=O)CCCCO)=O)cnc2n1CCOC2 40924,C1(C(=O)NCc2ncc[nH]2)(COC)CCCN1C(=O)CC(O)CN(C)C 40925,C(C(CC(F)(F)F)NC(=O)CCOC)NC(c1ccc(N(C(C)=O)C)cc1)=O 40926,c1(C(N2C(CNC(c3ncn(CC)c3)=O)CCC2)=O)cc2scnc2[nH]1 40927,CN1CCN(C(C2CCCCC2(F)F)=O)C(CNC(c2cc(O)ncc2F)=O)C1 40928,c1(C(=O)NC(CCC)C2CCC2)oc(CNC(C2(Cl)CCCCC2)=O)nc1C 40929,N1(C(C(C#C)(C)C)=O)CC2(CCN(C(C3(c4ccsc4)CC3)=O)CC2)C1 40930,N1(c2c(CC)c(Cl)ncn2)CCC2(CCN(C(=O)COCC(=O)N)C2)C1.C(C)=O 40931,C#CC1(C(=O)NC(COC)CO)CN(C(c2cnnn2C=C)=O)C1 40932,N1(C(=O)Cn2cc(CCCOCCO)nn2)CCOC(c2cccc(Cl)c2)C1 40933,c1(C(=O)NCCNC(=O)CCC2CCC2)cccc(F)c1 40934,N1(C(C(C)=C(CC)C)=O)CC2CC(C1)C2NC(=O)CN1CC(C)C1 40935,CC1CC2CC(C(=O)NCCC3CCCN(C(=O)C4=COCCO4)C3)(C2)O1 40936,c1(C(C)NCC2(NC(=O)OC(C)(C)C)CCCCC2)ccc(Cl)c(F)c1 40937,N1(C(C2C(C(=O)OC)CC2)=O)CCC(C(=O)NC(c2nc(C)no2)C)C12CC2 40938,C1(NC(C2(C(=O)OC(C)(C)C)CCC2)=O)CCOC(c2ccc(F)cc2)C1 40939,n1(CC(=O)NCC2(NC(C3CCCO3)=O)CCOC2)cc(F)ccc1=O 40940,CC1Oc2ccccc2OC1C(=O)NC1CCC2(CN(Cc3nncs3)C2)O1 40941,N1(C(C2(C(C)(C)C)CCCC2)=O)CC2CN(C(C3CCCS3(=O)=O)=O)CC2(C)C1 40942,CCCC(CCC)CC(=O)N1CCN(C(=O)COCCSC)C(CS(C)(=O)=O)C1 40943,C1(C(=O)NC(CNC(C(C(C)C)NC(=O)C(C)(C)C)=O)(C)C)CCC(F)(F)CO1 40944,C(=O)(C(C)(C#N)CC)NCc1c(CNC(c2c(CC)nn(C)c2)=O)cccc1 40945,N1(C(c2cc(C)c(Cl)cn2)=O)CCCC(C2CCN(C(=O)CCCC#N)C2)C1 40946,C(c1cncc(C)c1)=CC(=O)N(C(CN(C(C1(CC=C)CCCCC1)=O)C)C)C 40947,CC(C1CCCCC1)=CC(=O)NCC(C)NC(=O)Cc1cc(C)n(C)n1 40948,NC(=O)CC(C(=O)N1CCCC(C(F)F)C1)NC(c1ccc(O)cn1)=O 40949,CCC(C(=O)NCCC1CCN(C(=O)C(N2CCC(C)CC2)=O)CC1)C(C)O 40950,c1(C(N2CCC(NC(C(C(C)C)OCC)=O)C2)=O)cnc(C)nc1C1CC1 40951,N1(C(CC(C)F)=O)CCC(CNC(=O)CN(S(C)(=O)=O)C)C(F)(F)CC1 40952,N12CCCC(CCOCCO)(C1)OC(=O)C2.c12cnc(s1)C(=O)NC2.C1(C)CC1 40953,CC(C)(C)CCCCC(=O)NCCC1CCN(C(c2cc(F)c(F)cc2O)=O)C1 40954,C(C)(C)(C(=O)N(CCCNC(C1(C)CCCC1)=O)CC1CCC1)N(C)C 40955,N1(C(CNS(NC)(=O)=O)=O)CCCC(CNC(=O)Cc2cc[nH]n2)CC1 40956,CCCC(C)(C)C(=O)N1CC(C(=O)Nc2ccc(Cl)cc2O)CC(C)C1 40957,O=C(C1CNc2ccccc21)N1CCN(Cc2ccc(Cl)cc2)C(=O)C1 40958,C=CCC(CC=C)C(=O)NCCN(C)C(C1N(CCCC)CCC1)=O 40959,CS(=O)(=O)C(C(=O)NCCCNC(C1(F)CCCCC1)=O)C1CC1 40960,Cc1c(C(=O)NCCN(CCCN(C)C)C(=O)CC2CCC(O)C2)ncn1C 40961,Cc1nc(Cl)[nH]c(=NC(C)CC(C)NC(=O)CC2CCCC2)c1F 40962,CCCCC(CNC(=O)C1=CCCC1)NC(=O)CCc1cnc(C2(C)CC2)o1 40963,C1(C(N2CCCC(CC)C2)=O)C2CC3C(C2NC(=O)C(C)(O)CCOC)C13 40964,N1(C(C(C)=C2CCC2)=O)CCN(C(=O)CC(F)(F)Cl)C(C(C)C)C1 40965,c1(C(N(CC(C)NC(c2n[nH]cc2Br)=O)C)=O)cc2c(cc1O)CCC2 40966,C1(CNC(C2(C(C)NC(CCCOC)=O)CC2)=O)CCOC(C)(C)C1 40967,c1(C(N2CCC(C)(NC(C(C)OCCOC)=O)CC2)=O)ccc2occc2n1 40968,CN1CC(C(=O)NCC(C)(C)CN(C(=O)Cn2cnnn2)C)C(C(F)(F)F)C1 40969,c1(C(=O)NCCN(C(=O)CC2C=CCC2)CCC)c[nH]c(C)c(Cl)c1=O 40970,c1(CNC(CC)C(N)CO)cc(C(F)(F)F)ccc1F 40971,c1(C(=O)NC(CCNC(c2c(COC)nn[nH]2)=O)(C)C)cn2c(n1)CCCC2C 40972,c1(C2(C3CC3)CN2)nnnn1CCCOC.C1(CNC2(C)CCC2)CC2CC2C1 40973,c1(CC)ccc2occ(C(N3CCC(C)(CNC(c4cc[nH]c4C)=O)C3)=O)c2c1 40974,c1(C(=O)NC(CNC(C=NOC)=O)CO)cc(Br)c([N+](=O)[O-])[nH]1 40975,C1(NC(C2(N(C)C)CC2)=O)CCCC(N=c2[nH]c(Cl)nc3ncn(C)c23)C1 40976,C(=O)(CC1CCOc2ccccc21)NCC1C(NC(c2cnc(C)s2)=O)CC1 40977,c1(C(C)C)ncc(NC(=O)C(C)NC(=O)CC2CC2C2CC2)cn1 40978,CC(C)(C)C(C)(O)C(=O)N1CCN(C(=O)C2=CCCCCC2)C(CC(F)(F)F)C1 40979,N1(C(CNC(CC)=O)=O)CC(NC(=O)C(C2CC2)O)CC2(CCC2)C1.NCC 40980,c1(C(N2CCCC(CCNC(CC(=O)N(C)C)=O)C2)=O)cc(Cl)ncc1N 40981,CC1(C)CCC(C(=O)NC2(CNC(C3CCOC3)=O)CCOC2)C1 40982,C1(NC(COCCOC)=O)CC(C)CN(C(=O)C(c2c(OC)cccc2Cl)=O)C1 40983,CCN=C(NCC1CCCC1C(=O)NC(C)(C)C)NC(C1CCOC1)C 40984,C1(CC(=O)NCCCCN(CCCNC(C(CCC)C)=O)C)COC(C)(C)CO1 40985,C(=O)(CC1OCCc2ccccc21)NC1CC(NC(C2(C)CCC(O)CC2)=O)C1 40986,C12(NC(Cc3nc(CC)sc3)=O)CCN(C(=O)COC3(C)CCC3)CC1C2 40987,C12(C(N3C(CNC(c4c(C)onc4C4CC4)=O)CCC3)=O)CCC(CC1)C(C)O2 40988,C1(COC(C)(C)C)CCCN1C(=O)C(=O)NC1CCCC1CN 40989,C=CCC(CC=C)C(=O)NCC(CNC(c1cc(C2CC2)oc1C1CC1)=O)CO 40990,N1(C(=O)Nc2ccc(CC)cc2)CCCN(CC2C3CC4C(C3)C24)CC1 40991,C1(F)(CNC(CC2(CSC)CC2)=O)CC(NC(=O)C(C)(C)C2CCCCO2)C1 40992,c1(C(N2CC(C(C)NC(Cc3c(C)noc3)=O)OCC2)=O)ccn2nnnc2c1 40993,N1(SS(C)(=O)=O)CCN(C2CCCN(C(=O)CSc3ccccn3)C2)C(=O)C1 40994,c1(C(N2CC3(C(NC(c4ccc(F)s4)=O)CC3)C2)=O)coc2ccccc12 40995,c1(C(N2CCC(C)(CNC(CN3C(C)CC3)=O)C2)=O)cnc2[nH]cnc2c1 40996,CC(CNC(=O)CNC(=O)CNC(C1CC2CC2C1)=O)S(C)(=O)=O 40997,c1(C(=O)NCCOCCNC(CC(COC)(C)C)=O)cc(N)c2ncccc2c1 40998,c1(C2CC2SCCC(=O)NCCNC(C(C)(C)F)=O)ccc(F)cc1F 40999,C(C(CC(C)C)NC(=O)C(O)C(F)F)NC(CCCN(C(=O)OC)C)=O 41000,N1(C(CCOC)=O)CCC2C(C1)NC(=O)N2C1CCN(C(=O)CC(C)(C)C)CC1 41001,C=CCCC(C1CC1)NC(=O)C#CCNC(c1csc(Cl)n1)=O 41002,C1(NC(C2C(C)C2)=O)CCOCC1C(=O)NCC(=O)NC1CC1 41003,CC(C)CC(O)C(=O)NCC1CC1C(=O)NC1(CO)CC(F)(F)C1 41004,c1(C(=O)NC(C(CO)NC(COc2cccc(OC)c2)=O)C)ccc(C)nc1O 41005,C(=O)(C1=NN(C)C(=O)CC1)N1C(C)CCC(NC(c2csc(C(=O)O)c2)=O)C1 41006,N1(C(CC(=O)N(C)C)=O)CC(C2(NC(=O)CCc3ccoc3)CC2)C1 41007,CC1CN(C(=O)CSc2n[nH]c(O)n2)CCC1NC(=O)C(C)n1ccnc1 41008,c1(C(N2CCOC(CCNC(C3(CF)CC3)=O)C2)=O)ccc2cnsc2c1 41009,CC(C)C(O)C(=O)N1CCC(CCNC(C2(c3ccccc3F)CCC2)=O)CC1 41010,c1(C(=O)OCC2Cc3ccccc3CO2)n[nH]c2c1CCCCC2 41011,CC#CC1CN(C(C2(NC(=O)Cc3ccc[nH]3)CCCC2C)=O)C1 41012,N1(C(c2c(C#C)c[nH]n2)=O)CCC(C=C)(C(N2CCCC(OC)C2C)=O)CC1 41013,Cc1cc(C)n(CCCNCc2ccccc2-c2ccc(F)cc2)n1 41014,C(c1cc(Cl)ccc1Cl)=CC(=O)NC1C(NC(Cc2ccc(C)s2)=O)CC1 41015,C1(C(N2CCC(CCNC(C(CSC)O)=O)CC2)=O)CCc2ccccc2C1 41016,N1(C(C2(O)CCN(CC3CCOC3)CC2)=O)CCc2cccc(O)c21 41017,CCCC(CNC(=O)CSC(F)F)NC(=O)CCOCC 41018,c1(C(=O)NC2(CF)CCN(C(Cc3c(C)nc(C)s3)=O)C2)cc(C)c(F)cc1F 41019,C1(NC(c2cc(OC)c(F)cc2)=O)CCN(C(C2CC2(Cl)Cl)=O)CCC1CO 41020,Cc1c(C(=O)NCC(C2CCCCN2C(c2cnc[nH]2)=O)(C)C)cnn1C(C)C 41021,N(C1c2ccccc2CC12CCNCC2)CC1N(C(N)=O)CCC1 41022,N1(C(COCC)=O)CC(NC(=O)CC2(C)CC2)C2CC12 41023,N1(C(CC2CN(C)C2)=O)Cc2ccccc2CC1CNC(C1CC2C=CC1C2)=O 41024,N1(C(Cc2cnc(C)[nH]2)=O)CCOCC(C)(CNC(=O)C(C)NC(=O)C2CC2)C1 41025,CC1(C)C=C(C(=O)N2CCN(C(c3cnn(C4CCC4)c3)=O)C(C3CCC3)C2)C1 41026,N1(C(C2C(C)C2C)=O)CC2CC(C1)N(C(=O)CN1CCN(C)C(=O)C1)C2 41027,N1(C(C(CC#C)C2CC2)=O)CCC2CN(C(c3cc4sc(C)cc4s3)=O)CC12 41028,c1(C(N2CC3CN(C(C4(F)CCC4)=O)CC(C2)O3)=O)cc(Cl)cc(Cl)c1[N+](=O)[O-] 41029,CC(C)(CS(N)(=O)=O)C(=O)NCC1CN(C(C2(O)CCC2)=O)CC12CC2 41030,CN1CCC(C(=O)NC2(C)CCN(C(=O)CC3CCSCC3)C2)S1(=O)=O 41031,C1(C(=O)NCC2CCC(C(=O)NCc3cnc(CC)s3)O2)CC2CCC1O2 41032,CC(c1cccnc1)=CC(N1CC(NC(c2nccc(C)c2N)=O)C2(CC2)C1)=O 41033,Cc1cc(NC(=O)C#CCNC(C2COCCC2C)=O)cc(CO)c1 41034,CCC(CC=C)NC(=O)CC1(OC)CN(C(=O)CC2CCC(=O)C2)C1 41035,Cc1nc(F)ccc1NC(c1ccc(NCCC(C)C)cc1Cl)=O 41036,c1(CC(=O)NC(c2cn(-c3ccc(C)cn3)nn2)C)ccc2occc2c1 41037,c1(C(=O)NCCN(C(=O)C2=CSCCO2)CCC)c[nH]c2c(OC)nccc12 41038,C(=O)(CC(C)CC(C)C)NC(CC=CC)C(=O)NCCc1cccnc1F 41039,c1(C(=O)NC2CC(NC(C(C3CCCCC3)OC)=O)C2)cccc(C(F)(F)F)n1 41040,CN1CCc2[nH]nc(NC(N3CCOCC3CC(c3ccco3)O)=O)c2C1 41041,O=C(C1=Cc2cc(F)ccc2OC1)NCC1CC(NC(c2ccno2)=O)C1 41042,c1(OC)cc(NC(C2CCCN(C(=O)C(=O)c3ccco3)C2)=O)ccc1Cl 41043,C12(C(NOCCCC#C)=O)CCN(C(=O)CCOCCOCC)CCC1C2 41044,c1(C2C(C(=O)OC)C2)cccnc1-c1ccccc1N 41045,CC1CCCC(C)C1NC(=O)CCOCCCNC(c1ccc(CC#N)cc1)=O 41046,c1(NCC(CC)(C)OCC)[nH]cnc1C#N 41047,C=CC(CC)C(=O)NC1(CC(=O)N(C(C)COC)CC)CC1 41048,N1(C(C(C=CC)O)=O)CC2C(CNC(=O)CNC(=O)Nc3ccccc3)C2C1 41049,Cc1ccc(F)cc1CC(=O)NCCCC(C)NC(c1cnc(C)n1C)=O 41050,c1(C(=O)NCCCCC(C)NC(=O)C(F)(F)C(F)F)cnc2c[nH]nc2c1 41051,CC1(CC(=O)NC2(CCO)CCCCC2)CCCN1C(c1ccoc1)=O 41052,N1(C(C2=C(C#N)CCC2)=O)CCC2(CCC2)C(CNC(c2ccoc2Cl)=O)C1 41053,C1(CNC(c2cc(C(C)=O)sc2)=O)CN(C(c2ccc(O)nn2)=O)CC1C 41054,Cc1nc(C(=O)NC2CN(C(C3CCCN3C=O)=O)CC2C)c2ccccn12 41055,N1(C(CN(CC#C)C(c2cn(C)nc2CC)=O)=O)CCCC(CN(C)C)CC1 41056,N1(C(C2C(C(C)NC(C3(SC)CCC3)=O)C2)=O)CCC2(CC1)CC(O)C2 41057,C=Cn1nncc1C(=O)NCCCCCNC(c1c(Br)n[nH]c1C)=O 41058,C(=O)(CC(CC(C)C)NC(c1ncccc1CC)=O)N(C(C=C)C)C 41059,C(C)(CC(=O)N(C1CCN(C(C2(N(C)C)CC2)=O)C1)C)=C(C)C 41060,C(=O)(C(CCNC(C)=O)OC)NCC(COC)NC(c1nn(C)cc1N)=O 41061,c1(C(=O)NC2C(NC(CCN(CC(F)(F)F)C)=O)CC2)cccc(N)c1 41062,c1(CC(=O)N(CCCCCNC(C2(C#C)CCC2)=O)C)cccc(F)c1F 41063,C12(C(=O)NCCCC(C)(C)NC(C=CC(C)C)=O)C3C(=O)C4C5CC(C14)C2C35 41064,N1(C(Cn2cc(C(=O)OC)nn2)=O)CC2CC3CC2C1C3NC(=O)CSC(C)C 41065,Cc1cc(C#N)c[nH]c1=NC1CN(C(=O)CC(C)C2CCCCC2)C1 41066,c1(C(=O)NCC(CN(C(CCC(C)OC)=O)C)O)cc(N)c(Br)cc1C 41067,c1(C(=O)NC(C2CN(C(=O)CC3CCC(=O)N3C)C2)C)ccc2nc(O)[nH]c2n1 41068,Cc1[nH]nc2ccc(CN3CC4(C)CN(C(=O)CNS(C)(=O)=O)CC4(C)C3)cc12 41069,S(=O)(=O)(c1cccnc1NC(c1cnc(C)s1)C)N1CCC(OC)CC1 41070,C1(C(C)C)(C(=O)NCc2nocc2C(C)(C)C)CCN(C(=O)OC(C)(C)C)CC1 41071,C1(C)(NC(C(C)NC(N)=O)=O)CN(C(=O)C=CCN2CCOCC2)C1 41072,c1(C(C(=O)NC(C(CO)NC(C(CC)C)=O)C)(C)C)cccc(F)c1 41073,c1(C(N2CCC(NC(C3(C)COC3)=O)C2)=O)nccnc1Sc1ccccc1 41074,C1(CC)CN(C(c2cnn(C)c2CC(C)C)=O)CCN1C(=O)CS(=O)(=O)N(C)C 41075,c1(CC)oc(C)cc1C(=O)NCCC(C)N(C(=O)Cc1cc(C)cs1)C 41076,CC(C)CC(O)C(=O)NC1CCCN(C(c2cccc(C3(F)COC3)c2)=O)C1 41077,N1(C(=O)NC2CCCC(F)(F)C2)CCC2(CCc3ccccc32)C1 41078,C1(N(C(C(C)CC2CC2)=O)C)CCCN(C(=O)Cc2cncc(Br)c2)C1 41079,N1(C(C2C(NC(=O)CC3CSCCO3)COC2)=O)CCC2(CC1)CC(O)C2 41080,c1(CC(C)C)ccccc1CN(C)C(=O)NC(CCc1ccc(Cl)cc1)C(C)C 41081,c1(C(=O)NC2CC(OC)C2)cc(CCNC(c2c[nH]c(=N)o2)=O)on1 41082,C1(NC(c2c(C)n(C3CC3)nc2)=O)CC2(CCN(C(C3(C)C=CCC3)=O)C2)C1 41083,C(=O)(C1=C=CCCCC1)NCC(CNC(C1CCC(=O)NC1)=O)F 41084,c1(OC)ccc(CC(=O)NC2CCCC(CN(C(=O)CCC(N)=O)C)C2)nc1 41085,Cc1ccc(OC(C)C(N2CC(NC(=O)C(C)N(C)C)C(C)C2)=O)cc1 41086,N1(c2ncc(C)c(O)n2)CC(CNC(C2(C)CCCCO2)=O)OC(C)(C)C1 41087,N1(C(=O)COCC2CCCO2)CCC2C(C1)CN2C(c1cc(CC(=O)O)c[nH]1)=O 41088,c1(OC)nccc(C(=O)NC2CC(NC(C3(OC)CCC(C)C3)=O)C2)n1 41089,N1(CC(C#C)C2CCC2)CCCC1(C)C 41090,c1(CNC(C2C(CCC)C2)=O)nnn(C)c1C(N1CCC(OC2CCC2)C1)=O 41091,Cc1cc(F)c(C(N2CCC(NC(c3ncccn3)=O)C(C)C2)=O)cc1F 41092,C1(C#N)(C(=O)NCCCCCCNC(CC2C(C)CCO2)=O)CCCCCC1 41093,CCC(C)CCCCC(=O)N(C)CC1C2CN(C(=O)C=C(C)C(C)C)CC12 41094,c1(C(=O)NC2C(NC(c3cc(C)c(Cl)s3)=O)CC2)cccc2nn(C)cc12 41095,C1(C(=O)NC(C#C)(C)C2CCOC2)CN(C(=O)CCC2CCC(=O)C2)CC12CC2 41096,c1(CCCC)ncc(C(N2CC(C(N)=O)(CNC(=O)CC3CN(C)C3)C2)=O)s1 41097,c1(C(=O)NC(C2CCCN(C(c3n(CC)ncc3)=O)C2)C)cc2n(c1)CCSC2 41098,c1(C(=O)NC2C(NC(c3cc(C4CCC4)on3)=O)CCC2)ccn2ccsc12 41099,c1(C(N(CCC(=O)N(C)C)C(C)C)=O)cnc(O)c2cncn12 41100,c1(C(=O)NC2C(NC(C(COC)NC(C)=O)=O)CC2)ccnnc1C 41101,C=C(CNC(=O)C(CCC1CCC1)NC(C1CC(=O)C1)=O)C(F)(F)F 41102,Cc1ccccc1C1(C(=O)NCC2CC(NC(c3n[nH]cc3Cl)=O)C2)CC1 41103,C1(CNC(COCCCC)=O)CN(C)CCN1C(c1cc(C2CC2)nc(O)c1)=O 41104,N1(C(C2(F)CN(C(c3cc(C)no3)=O)C2)=O)CC2CCC2(C)C1 41105,c1(C(=O)NCC2C3CN(C(CC(=O)NC4CC4)=O)CC32)ccc2scnc2c1 41106,N#Cc1ccc(S(=O)(=O)N2Cc3ccc(O)cc3C2)nc1 41107,c1(C(=O)NCC2(F)CC(CNC(=O)CC3CCC4CC34)C2)cccn2nncc12 41108,Cc1[nH]c(C#N)cc1C(N1CCC(C)(CC(=O)NCCN2CCNC(=O)C2)C1)=O 41109,C1(C(N2CCC(N(C(c3cc(C)n(CCO)n3)=O)CC)C2)=O)C(C)OC(C)C1C 41110,C(C(C(C)C(C)C)NC(=O)C(C)(C)O)NC(c1c(OC(C)C)cccc1)=O 41111,c1(C(N(CC(CN(C(CCOC(C)C)=O)C)O)C)=O)cn(C)cc1C(F)(F)F 41112,c1(OC)cccc2c1OCC(C(=O)NCC1CCCN(c3nccs3)C1)=C2 41113,c1(C(=O)NCCC2(C(=O)NCc3c(C)occ3)CCC2)cn(C)c(C)n1 41114,c1(C(=O)NCCCCNC(C(C)(C)OC(C)=O)=O)snc(Cl)c1Cl 41115,C1(NC(c2cncc(SC)c2)=O)CCCN(C(C2(S(C)(=O)=O)CC2)=O)CC1 41116,C(=O)(N=c1[nH]nc(-c2ccc(OC)cc2)s1)N1C(CC(C(=O)OC)F)CC1 41117,C1(O)(C(NCc2c(COC)ccs2)C2CC2)CCCC1C 41118,O=C(CCCn1cncn1)NCCCc1cn(C2CCCC2O)nn1 41119,C(CC1=CCCCCC1)NC(CC(CC#C)NC(c1ccc(C2CC2)o1)=O)=O 41120,C1(OCCNC(CN(CCOC)C)=O)CCN(c2ncns2)C1 41121,Cc1nc(C(=O)NCC2(C)CCC(NC(=O)CCC(=O)N(C)C)C2)c(C)n1C 41122,C1(O)(CNC(C2CC(CCC)C2)=O)CCCN(C(=O)COC(=O)CO)CC1 41123,CC1(C(=O)NC2CCC(C(=O)NC3CCOCC3F)C2)CC2C=CC1C2 41124,C#CCC(CC#C)C(=O)N1CC(CNC(c2cncc(C)n2)=O)C2CC12 41125,C1(CCOC)(NC(c2c(CCC)[nH]cc2)=O)CCN(C(=O)C(C)(C)CN(C)C)C1 41126,C1(NC(=O)C#CCNC(=O)CC2CCC(=O)C2)CCN2CCCCC12 41127,C(CCC(C)NC(c1cscc1OCC)=O)NC(CN(S(CC)(=O)=O)C)=O 41128,N1(C(C(N2CCC(CC#C)CC2)=O)=O)CCC2(CC1)CC2C#N 41129,N1(C(COC)=O)CCN(C(=O)CNC(c2cccs2)=O)C(C)CC1C 41130,c1(OCC=C)cc(Cl)ccc1C(=O)NC1CC(NC(C2(C3CC3)CC2)=O)C(O)C1 41131,c1(CCN=C(NCCSC)NCC2CCN2C)c[nH]c2ccccc12 41132,c1(NCC2N(Cc3nc(C)sc3)CCC2)ccc(C(N)=O)cn1 41133,C1(NC(c2c(C)oc(C(C)C)c2)=O)CCCN(C(c2[nH]nnc2C2CC2)=O)C1C 41134,CC(C)(C)C(CC(=O)NC12CCOC(CNC(=O)CN3CC=CC3)(C1)C2)C(F)F 41135,Cc1cc(C)cc(C=CC(=O)NCC(CNC(C2C(C#N)C2(C)C)=O)CO)c1 41136,C(=O)(C1=CCCC1P(C)(C)=O)N1CC(C)C(NC(c2cc(C3CC3)ccn2)=O)C1 41137,c1(C(=O)NC(C)CN(C)C(C2CCN(C)C2)=O)cnc2ncc(Br)cc2c1 41138,N1(C(CCC2CC(OC)C2)=O)CC(NC(=O)C(N2CCCCCC2)C)CCC1C 41139,CC(C)(C)C(CO)C(=O)N1CCN(CCNC(C2CCn3ncnc3C2)=O)CC1 41140,N1(C(c2c(C)ccn2C)=O)CCC2(CC1)CN(C(=O)C1=CCCCC1C)C2 41141,C1(CN2C(=O)NC(c3cc(F)cc(F)c3)C2=O)CC2(C1)CC(F)(F)C2 41142,c1(NC)cc(Cl)ccc1C(N1CC2(NC(=O)CC3(OC)CCC3)CCC1C2)=O 41143,c1(C(N(CC#C)C)=O)cc(CNC(C2CC(F)(F)C2)=O)no1 41144,CCC(C)CC(=O)C(=O)NCC(C(=O)NCCC(C)(C)C1CC1)C(C)(C)C 41145,C(c1ccccc1C)=CC(=O)NC1(C(=O)NCC(CC)O)CCSC1 41146,N1(C(CCOc2c(C(C)C)cccc2)=O)CC(NC(C2CC2F)=O)CCC1C 41147,c1(C(N2C(CNC(c3cc(C(=O)OC)on3)=O)CC(O)C2)=O)ccc([N+](=O)[O-])[nH]1 41148,C1(n2cc(C(=O)NCc3c(OCC=C)cccc3)nn2)CCCC1S(C)(=O)=O 41149,c1(Cn2ncc(C(N(CCN(C)C(C3CC3Cl)=O)C)=O)c2)ccccc1Cl 41150,CC1CCN(C(C2CCCN(C(N)=O)C2)=O)CC1NC(=O)C(F)n1cccn1 41151,N1(C(C(CC)=O)=O)CCC(O)(c2cn(C(c3ccccc3F)C)nn2)CC1 41152,c1(NCCC(N2CC3C(NC(C=CC=CCC)=O)(C3)C2)=O)oc(C)nc1C#N 41153,C1(NC(=O)OC(C)(C)C)CCOC(C(=O)NCc2cccn2C(F)F)C1 41154,N1(C(CC(c2cccc(OC)c2)C)=O)CCCC(N=c2nc[nH]s2)C1 41155,c1(C(=O)NC2COCCC2NC(C2(C3CCCO3)CC2)=O)cc2n(c1)CCCC2 41156,c1(CC)oc(C)cc1C(=O)NCCC1CN(C(c2ccc(OC)nn2)=O)C1 41157,CC(C(=O)N1CC(F)CC1C(=O)Nc1ccc2c(c1)CCO2)C(F)(F)C(F)F 41158,C(=O)(C1CS(=O)(=O)c2ccccc21)NC1(C)CCN(C(=O)C(F)(F)F)C1 41159,c1(C(C(=O)N(CC(C)C#N)C)NC(=O)C(F)C2CCC2)cn(C)nn1 41160,C1(C(N2CC(COC)(NC(=O)CC#N)C2)=O)CC2CCC1CC2(F)F 41161,N1(C(CN2N(C)C(=O)C2)=O)CC(O)(C2(CNC(=O)CNc3ccccn3)CC2)C1 41162,C1(C(=O)NCCNc2csc3nnsc23)CCC2(CN(C(CCCCC)=O)C2)O1 41163,c1(C(=O)NCC(C)(C)NC(C2C(C)C2C)=O)cc(C(F)(F)F)ccc1N 41164,Cc1ccc2c(c1)CCC2C(=O)NCC(CC(F)(F)F)NC(=O)CCCCCF 41165,C(CC(C)C)(C(=O)Nc1ccc(-c2ccno2)cc1)OC.C1C(=O)NNC(=O)N1 41166,c1(C(=O)NCC(CC(=O)NCC(C(C)(C)C)OC)(C)C)ccc2nccn2c1 41167,C1(CC=C)(C(=O)N(CC)Cc2ccccc2)CCCN1C(=O)CC1CSCCO1 41168,c1(C(=O)NC(CN(C(C2CN(C)C(=O)N2)=O)CC)C)nc(C)sc1Br 41169,c1(C(N(CCOCCC(=O)NCC=CC(=O)OC)C)=O)cc(OC)nn1C 41170,n1(CC)ncc(CNC(C2(OC)CCN(C(=O)Cc3cncnc3)C2)=O)c1C 41171,C=CC1(C(=O)NC(c2cccc(O)c2)C)CCN(C(c2[nH]ccc(=O)c2C)=O)C1 41172,c1(OC)nc(C)ncc1C(=O)NCC(C)NC(C1CCC2CC2CC1)=O 41173,C1(CNC(=O)C=Cc2ncc[nH]2)C2CCC1CN(C(C1CCCN1C=O)=O)C2 41174,C1(OC)CCCCC1CC(=O)NCCC1CN(C(c2cncnc2C(C)C)=O)C1 41175,N1(C(c2cncc(OC)c2)=O)CC2CCC1C2NC(=O)CS(=O)(=O)N(C)C 41176,Cc1cc(F)cc(NC(C2CC2NC(=O)CCCn2ccnc2)=O)c1Br 41177,C1(NC(c2n(CC)nnc2)=O)CN(C(c2ccc(C)cn2)=O)CC1N=[N+]=[N-] 41178,C(=O)(CC(C)CC(C)C)N1C(CNC(c2n(C(CC)CC)ncc2)=O)CC1 41179,C1(NC(C23C(C)(C)OCC2C3)=O)CCCC12CN(C(c1coc(C(F)F)n1)=O)C2 41180,CN1CC(O)CC1(C)C(=O)NCC(N1CCN(C(=O)C(=O)N(C)C)CC1)C(F)F 41181,CCCC(CC1CCCC1)C(=O)NCC(C(C)(C)C)NC(=O)CSCC(N)=O 41182,Cc1ocnc1C(=O)N(CCCCN(C)C(C1CCCC1c1ccccc1)=O)C 41183,C1(NC(CC(C=C)CC)=O)CCSC12CN(C(=O)C(CC(C)C)N(C)C)C2 41184,C1(C(C(=O)N(CCOC(C)=O)C)C)CCN(C(c2c(C)noc2C(C)C)=O)CC1 41185,CC1C(NC(C2CC3(CC3)CO2)=O)CCCN1C(=O)CCNS(C)(=O)=O 41186,C#Cc1cnc(NC(c2[nH]c(C)c(C(=O)NCCNC(C)=O)c2C)=O)cn1 41187,C1(c2cn(C3CCN(C(CN(c4ccccc4)CC)=O)C3)nn2)COC(C)(C)O1 41188,Cn1ncc2nc(Cl)nc(NCC3CN(C(C4CCS(=O)(=O)C4)=O)CC3(C)C)c12 41189,C1(C(N)=O)CCN(C(c2cccnc2CNC(=O)COc2cccnc2)=O)CC1 41190,C(CN=c1[nH]c2c(c(=NC3CCCc4ccc(F)cc43)[nH]1)SCC2)NC(=O)NC 41191,C(CC(C)(C)C(=O)NCCC(C)CCNC(c1cncc(N(C)C)c1)=O)SC 41192,Cc1[nH]nc(C(=O)NCC2CC(NC(c3ncccn3)=O)C2)c1C 41193,Cc1ncnc(C(=O)NCc2ccc(CNC(=O)C(C)C(C)O)c(F)c2)c1C 41194,c1(CCC(=O)NC23CN(C(C4CCN(C)C4)=O)C(C2)C3)ccc(Cl)cc1Cl 41195,N1(C(CCC#N)=O)CCC2(CCCC2NC(C2COCCC2(F)F)=O)CC1 41196,N1(C(c2cnc(CCC)s2)=O)CCCC(CCC)(NC(c2nccn2C)=O)C1 41197,N1(C(C2CCCS2)=O)CCOC2(CCC(N=c3[nH]c4ccc(F)cc4s3)CC2)C1 41198,C1(C(=O)NC(C2(O)CCN(C(C(C)(C)OC(C)C)=O)C2)C)CCCCC12CCC2 41199,N1(C(C(c2ccc(Cl)s2)C)=O)CCN(C(=O)COCC(C)(C)C)C(CC2CC2)C1 41200,C1(C(=O)NCC(CC)(C)NC(c2cc([N+](=O)[O-])n[nH]2)=O)CC2CC1CC2(F)F 41201,C1(N(CCC)CCNC(C)CCCCCC=O)CCc2ccccc2C1.OC 41202,C(CN=c1[nH]c(=NCCOC(F)F)[nH]c2c1COC2)(c1ccccc1Cl)N(C)C 41203,CC1CNC(=O)CN1C(C1(NC(c2coc(C(N)=O)c2)=O)CC(F)(F)C1)=O 41204,C1(CN(C)C(C2(C3CC3)CC2)=O)CCN(C(=O)CCCC2OCCO2)C1 41205,C1(C(=O)NC2CCN(C(CCOC)=O)C2C(C)(C)C)CN(C)C(=O)CCO1 41206,C1(CCC)CN(C(c2ccnc(S)c2)=O)CC1NC(c1cn(C)c(C)n1)=O 41207,CCC(CC)(CCNC(=O)C(F)C(C)C)NC(c1ccc(C2CCC2)cc1)=O 41208,Cc1ccnc(O)c1C(=O)NCCCC1CN(C(C2CCNC(=O)C2)=O)CCO1 41209,C1(C(=O)NCC(n2cc(-c3cn[nH]c3)nn2)C)CCCN1S(C)(=O)=O 41210,Cc1ncc(CCC(=O)N(CC(C)(C)CNC(C2CC2F)=O)C)s1 41211,Cc1coc(C)c1C=CC(=O)N(CCCNC(C1CC=CCO1)=O)CC1CCCC1 41212,C1(N(C(C2CC(CC)C2)=O)C)CCCN(C(=O)CCC2CCC(=O)NC2)CC1 41213,Cn1nccc1CN1CSCC1C(=O)NOCC(=O)OC1CCCC1 41214,c1(C(N2CC(COC)(NC(=O)C(=O)N(C)C)C2)=O)cc(N)c(C)cc1C 41215,CCC(C)C(C(=O)NC1CCCC1CNC(=O)CCCOC)N(C)C 41216,CN1CCC(C(N2CCN(C(=O)C=Cc3cnccn3)C(C3CC3)C2)=O)CC1=O 41217,C1(NC(C(C)=CC)=O)COC2C(NC(c3cnn(C)c3C(C)C)=O)COC12 41218,Cc1c(C(=O)NC2(CCNC(=O)CCn3cncn3)CCC2)cnn1CC(F)F 41219,CCCC(C)(C)CC(=O)NCC1CCN(C(C2C3CCCOC23)=O)C1(C)C 41220,c1(C(=O)NCC(CN(C(CCOCCOC)=O)C)C)c(O)nnc(C)c1C 41221,CC1(C)CCC(C(N2CC(C(N)=O)(CNC(=O)CCC3CCCCO3)C2)=O)OC1 41222,c1(C(=O)NCC(N(C(C(CC)(C)O)=O)C)C2CC2)cc(Br)ccc1C1CC1 41223,C(=O)(CC1=CCCCC1)N1C(C(C)NC(=O)C2=CSCS2)CCCC1 41224,c1(CN2C(C(=O)NC3CCN(CCCC)CC3)CC(F)C2)cc(Cl)c(O)c(Cl)c1 41225,CC1C(NC(=O)Cc2csc(Cl)c2)CCN1C(=O)CCc1cccs1 41226,c1(CC)ncc(C(N2CCC(CCN(C)C(c3ncccn3)=O)CC2)=O)c(C)n1 41227,C1(CNC(C2CCC(O)C2)=O)CC2(CCN(C(=O)C=C(Cl)Cl)CC2)CO1 41228,C(=O)(C(C(C)C)c1cccnc1)NC1CC(F)(CNC(C(CSC)OC)=O)C1 41229,N1(C(c2cc(CCC)[nH]n2)=O)CCC(C)(NC(=O)CCCOC(C)(C)C)C1 41230,c1(OCCC)ccc(Br)cc1S(=O)(=O)NCc1ccc(C2CCC2)cn1 41231,c1(N(C)CC2CCCO2)nnc(-c2ccccc2Br)n1CCN1CCCS1(=O)=O 41232,C1(CCCC)CCN(C(=NCCC(C)=O)NCC(C)(F)F)C1 41233,C(=O)(CCCC(=O)OC(C)(C)C)NCCC(C)CCNC(C1CC(=O)N(O)C1)=O 41234,C(=O)(C1=C(Cl)CC1)NC1(C)CN(C(C(C)CC2CC2)=O)C1 41235,C1(C(=O)NCCC(C)(C)NC(=O)C(F)=CC2CC2)CC(C(C)(C)C)=NO1 41236,c1(N(CCC(C)O)C)nc(=NCCc2ccns2)[nH]c2c1SCC2 41237,C1(C(C)C)N(C(=O)N(c2ccncc2Br)C)CC12CCC2 41238,c1(CN(C(C=COCC)=O)c2cccnc2)ccc(F)cc1O 41239,CC1CC(=O)NC1C(=O)NCCCNC(=O)CCOc1cccc(Cl)c1 41240,c1(C(=O)NCC2CCN(C(C3(C)ON=C(C)C3)=O)CC2O)cc(F)c(F)cc1O 41241,c1(OC)cc(C(=O)NC2CCC2NC(=O)COC(c2nccn2C)C)cc(C)n1 41242,C12(C(=O)NCC(CNC(CCCOC(C)C)=O)F)CC3CC(F)(C1)CC(F)(C3)C2 41243,C(=O)(C1=C(C)OCC1)NC(C(N1C(CC)CCC1)=O)CN(C)C 41244,CC1CCCC(CN2CCC(NC(N3CCN(C(c4cccs4)=O)CC3)=O)C2)C1 41245,N1(C(C(C2CCCO2)OC)=O)CC(O)(CNC(C2(C(F)F)CCC2)=O)C1 41246,c1(CC)n[nH]c(CC)c1CC(N1CCC(N2CCN(CC(C)O)CC2)C1)=O 41247,Cn1ncc(S(C)(=O)=O)c1C(=O)NCCNC(c1cnc2ccccc2n1)=O 41248,C1(C(=O)NCCN(C(=O)CN(c2ccc(Br)cn2)C)CC)COCC(C)(C)O1 41249,C1(C(=O)NC2C(n3cc(CCSC)nn3)COC2)CCCC(F)C1 41250,Cc1cccc2nc(C(N3CC4CCC(C3)N(C(=O)C=CS(C)=O)C4)=O)cn12 41251,C1(NC(C(C)SC)=O)CC(C(=O)NOCC(F)F)C1(C)C 41252,C1(CC(=O)N(C2CCCC2)CCNC(CC(C)N(C)C)=O)CCNC(=O)C1 41253,N1(C(c2c(C)con2)=O)CC2COCC2(C(=O)NC(C)CC2CCC2)C1 41254,C(=O)(CCCCCS(N)(=O)=O)N1C(C(C)(C)NC(C(C)O)=O)CCC1 41255,c1(C(=O)NCC2(C)CC(NC(C(CC)SC)=O)C2)oc2c(C)ccc(C)c2c1C 41256,C(CC(O)C(=O)Nc1cccc(NC(C2CCC(=O)N2C(C)C)=O)c1)SC 41257,CCCCC(CNC(=O)NCC)N(C)C(C1CCNCC1C)=O 41258,C1(C(N2C(C)(C(=O)NC3CCCC(COC)C3)CCC2)=O)CC2(CC(=O)C2)C1 41259,c1(OC)ccc(CCC(=O)NC2CCC2NC(=O)COc2ccc(F)cc2)cn1 41260,N1(C(c2nn(CC)c(=O)cc2)=O)CCOC2CCN(C(C3(O)CC3(C)C)=O)CC12 41261,N1(C(C2(C)CCCCC2)=O)CC2(CNC(C3CC(F)(F)C3)=O)CC1CO2 41262,CC1C(=O)CCC1CC(=O)NC1(CCNC(c2coc(C3CC3)n2)=O)CCC1 41263,N1(C(C=CCN(CC(F)(F)F)C)=O)CC(F)(c2ccncc2)C1 41264,C1(C(=O)NCC2(C(=O)OC)CCCC2)CC(F)CN1C(c1cc(F)c[nH]1)=O 41265,C1(C(N2CCCC(C)(NC(c3cc[nH]n3)=O)C2)=O)CC2(C1)CC21CCC1 41266,C1(NC(c2ccc(C(F)(F)F)cn2)=O)CC(CNC(C2CC(O)C2)=O)C(O)C1 41267,c1(C(=O)NC2CC(NC(C3C(CC(C)C)C3)=O)C(O)C2)c[nH]c2c(C#N)cccc12 41268,c1(-c2nc(C(C)CC(F)F)n(C3CSC3)n2)ccc(Cl)cc1O.C1(C)CC1 41269,Cc1cc(=NC(=O)c2cc(CNC(=O)C(C3CCCCC3)O)no2)[nH]n1C 41270,N1(C(C(C)=C(CC)C)=O)CCN(C(C2CCN(CCC)CC2)=O)C(C(C)C)C1 41271,c1(CC)cc(F)ccc1CC(=O)N(CC(O)CNC(=O)C1=COCCO1)C 41272,Nc1cc(C(=O)NCC(CO)NC(=O)CC2CC3CC3C2)cc(C(F)(F)F)c1 41273,CCC1=C(C(=O)N2CCCCC2CCCNC(=O)CCCOC(C)=O)CCCO1 41274,C(C(CC1CC1)C(=O)Nc1cscc1C1CC1)NC(C(C)Cn1ccnc1)=O 41275,CCC(CC)C(C)C(=O)NCCOC1CCN(C(c2csc(C(=O)OC)c2)=O)C1 41276,N1(C(C(C)=C(CC)C)=O)CC2(NC(=O)CCc3cccc(Cl)c3)CC1C2 41277,Cn1ccc2ccc(C(N3CCC4(CCCC4NC(=O)C=C4CCC4)C3)=O)cc12 41278,c1(NC(CC2N(C(c3c(C)ncnc3)=O)CCC2)=O)cnc(Cl)c(Br)c1C 41279,C1(NC(C(C)=C2CC2)=O)CCC2CN(C(C3CCCOC3C)=O)CC2C1 41280,N1(C(C(C(C)C)S)=O)CCCC2(C1)CN(c1ccnc(Br)n1)CCO2 41281,C(=O)(C(C)S(=O)(=O)CCC)NC1C2CN(C(c3cn(CC=C)nc3)=O)C(C2)CC1 41282,CC(=O)CCCCCCC(=O)NC1CCCC(NC(=O)C(C)CO)C1 41283,c1(C(=O)NC2CC(CNC(Cc3n(C)nnc3)=O)C2)cccc(-c2ccoc2)c1 41284,CC1(C)C(NC(=O)C2=C(Cl)CCC2)CCN1C(=O)CCC1CCCO1 41285,N=c1[nH]c2c(s1)CN(C(=O)Oc1ccc(Br)c(C(F)(F)F)c1)CC2 41286,c1(-c2cc(NC(C3CC(C(=O)OC)C3)=O)sc2)ccc(NC(C)=O)nc1 41287,C1(NC(C(C)NC(=O)OC)=O)CC=C(C(=O)Nc2cnc(C(C)C)nc2)C1 41288,C1(C(=O)NCC(CC(F)(F)F)NC(C2(CC)CC2)=O)CCCC2(CCC2)C1 41289,C#Cc1cccc(C(=O)NCC2CC23CN(S(=O)(=O)CC2CCC2)C3)c1 41290,CC1CN(C(c2cn(CCNC(C3CNC(=O)N3)=O)cn2)=O)CCO1 41291,C1(NC(C2OCC(C)C2)=O)CCCN(C(c2cnn(C(F)F)c2)=O)CC1 41292,c1(C(N2CCCC(O)(CNC(C3(O)COC3)=O)C2)=O)cc2n(n1)CCOC2 41293,CCC(C)CCC(=O)N1CCC(CC(=O)NCC(F)C(C)(C)O)C1(C)C 41294,n1(C(C)N)cc(-c2noc(C3CCCN3C(=O)OC(C)(C)C)n2)cn1 41295,C(=O)(C(C)S(=O)(=O)c1ccc(F)cc1)N1CC=C(CCCOC(=O)NC(C)C)CC1 41296,c1(C(=O)NCCC2(CNC(=O)CC3CCOC3=O)CC2)cnc2ncnn2c1O 41297,N1(C(C(N2CC(C(C)NC(=O)CCc3nc(=N)[nH][nH]3)C2)=O)C)CCN(C)CC1 41298,C1(C)(N(CCN(CC(C)C)C(C)=O)C)CCCO1 41299,N1(c2c(OC)c(Cl)ncn2)CCC(C2CC2)(CNC(c2cnoc2C(C)C)=O)C1 41300,C1(OC)CCC2(C(=O)NC(C)(C)C(=O)NC(Cc3ccco3)CO)CC12 41301,N1(C(c2c(C)nsc2)=O)CCN(C(c2cccc(-c3cnco3)c2)=O)C(C#N)C1 41302,N1(C(c2cccc(Cl)c2C(F)F)=O)CC2(CCC(CNC(C3CC34CC4)=O)O2)C1 41303,N1(C(c2c(C)c(N)cnc2)=O)CC2CC(NC(=O)CC3(N(C)C)CCC3)C(C2)C1 41304,c1(NC(C(C2CC2)NC(c2ccc(OC)cc2)=O)=O)cc(C)ccc1C 41305,c1(C(=O)NC2CN(C(C(C(C)C)OC)=O)CC2SC)cncc2c(O)nccc12 41306,C1(N(C(=O)CSCC2CCCCO2)CC)CCCN(C(=O)C(C)(C)O)CC1 41307,N1(C(CS(N)(=O)=O)=O)CCC(CN2C(=O)CNC2=O)CC12CC2 41308,C1(O)(CN(C(C(CCC)O)=O)C)CCN(C(c2cc(C)c(CC)s2)=O)CC1 41309,c1(C(N(C2CC(NC(c3c[nH]ccc3=N)=O)C2)C)=O)ccc2c(c1)CCO2 41310,N(C(=NCCN1CCCC1)NCC1CCCC1C)Cc1c(OCF)ccc(Cl)c1 41311,N1(C(c2cnn(CCOC)c2C)=O)CCC2(CCN(C(c3ccc[nH]3)=O)C2)C1 41312,C1(CNC(C(=O)N(C)Cc2ccc(CO)cc2)=O)CCC(C)(C)CC1 41313,CC1CCN(C(c2sccc2C2CC2)=O)C(CNC(c2cc(=O)cc(Cl)[nH]2)=O)C1 41314,C(CCC(=O)NCc1nocc1C(=O)NC1CCCSC1)OC(C)=O 41315,c1(C(N2CC(CNC(CCCCOC)=O)OCC2)=O)nc2c(s1)COCC2 41316,c1(CC)ccc(C(=O)NC2(CNC(c3cnn(C)n3)=O)CCCCC2)cc1N 41317,C(=O)(C1=CC2CCCCCC12)N(CCNC(CS(C(C)(C)C)(=O)=O)=O)C1CC1 41318,c1(C(=O)OCC)sc(NC(=O)C(=O)N(CCCN2CCCC2)CC)c(C#N)c1C 41319,Cc1cc(C(=O)NC2CCC(N3CCOCC3)C2)nc(C)c1 41320,N1(C(C2(c3cccc(C)c3)CC2)=O)CCN(C(C2CC3(CSC3)C2)=O)CC(O)C1 41321,c1(OC)ncc(-c2nc(C)c(NC(c3nccc(Cl)c3Cl)=O)s2)cc1C 41322,C1(C(=O)NC2CC(NC(CN3CCC(C)CC3)=O)CC2O)SC2C=CC1CC2 41323,N1(C(C(C)n2cccn2)=O)CCOCC1(C)c1cn(CCSC2CCOC2)nn1 41324,C(=O)(N=c1[nH][nH]c2cc(C#N)ccc12)c1n(C)cc(NCc2ccnc(Cl)c2Cl)n1 41325,c1(NC(C2(C)CCN(C(c3cccc(F)c3F)=O)C2)=O)cc(Br)cnc1Br 41326,C12(NC(C(CSC)C)=O)CC1CN(C(=O)Cc1ccnn1C)C2 41327,N1(C(c2ccc(CC)nc2)=O)CCN(C(=O)C(C)=C(C)C)CC1c1ccnn1C 41328,c1(C(=O)NC2C(CNC(=O)CCC3CCCC(=O)N3)C2)cccc2[nH]nc(O)c12 41329,C(CCC(=O)N1CCCC1C(C)(C)NC(C1C=CCCC1)=O)N(C(=O)OCC)C 41330,CCC(CCC(=O)N(C1C2CN(C(c3cncn(C)c3=O)=O)CC12)C)NC(C)=O 41331,C(c1cc2ccccc2o1)=CC(N1CC(CCNC(C(C=C)(C)C)=O)C(C)C1)=O 41332,C(CCCC(CO)NC(C1(N2CCCC2)CC1)=O)NC(CC(CC)SC)=O 41333,CCCCCC(F)C(=O)N(CCC(C)(C)NC(c1ccsc1)=O)C 41334,C=CCC(C)(C)C(=O)N1CCCOC(CNC(C2CC2C(C)O)=O)C1 41335,C1(C(N(CCC(=O)NC(C)CCN(C)C)CC)=O)CCCSC1 41336,c1(CC)sc(C(=O)NC(C)CCNC(c2nnsc2C)=O)cc1Br 41337,C1(C(=O)NC2CC(NC(c3c(CC)cccc3CC)=O)C2)CN2CCN1C(C)C2 41338,CC1(CNC(=O)Cc2ccoc2)CC(NC(=O)Cc2cc(Br)cs2)C1 41339,N1(C(C(C)C2CCCC2)=O)CC2CC(NC(C3(C)COC3)=O)CC1C2 41340,C(CSC)(C(=O)NCc1cc(C(=O)NCC(C(C)C)OC)no1)OC 41341,C1(C(N(CCCCNC(c2cc(C)c(O)nn2)=O)C)=O)CCc2ncsc2C1 41342,C(=O)(CS(=O)CCC(F)(F)F)NC1CN(C(CCCCC(N)=O)=O)CC(F)C1 41343,C=CCCCCC(C(=O)NCc1cccc(Br)c1)N1CCC(O)C(C)(O)C1 41344,O(NC(=O)CC(CC=C)NC(C1CCOCC1)=O)CCOCC#C 41345,c1(C(c2ccc(C)o2)NC(C(C)(C2CC2)OC)C)ccc(S(N)(=O)=O)cc1 41346,CC1CN(C(=O)CCN2CCC2)CCCN1C(=O)C=CC(c1ccc(F)cc1)=O 41347,c1(CC)ncsc1C(=O)NC(C)(CNC(C1CCCC1CF)=O)CO 41348,C1(CC(=O)OCC)NC(=O)N(CC(C)OC(F)F)C1=O 41349,C12(CNC(C3N(C)CCCC3)=O)CCC(CC1)CN2C(c1cc(Cl)cnn1)=O 41350,C(=O)(C1=C(Cl)CCOC1)NC1CCN(C(CCC2C(C)=NOC2=O)=O)C(C)C1 41351,CC(C)C(C(=O)NCC1CN(C(C23CCC(C2)OC3)=O)C1)n1cccc1 41352,C1(C(=O)NC(CCC)C)OCCC1NC(=O)CCC1CC(OC)C1 41353,C1(NC(CSC)=O)CCN(C(c2ccc(CCO)cc2)=O)C1C 41354,N1(C(=O)OC(C)(C)C)CC2CCC1C2C(N1CC(CNC(=O)C(N)=O)C(C)C1)=O 41355,C1(C(=O)NCC(c2cccc(F)c2)C)CC2CC1CN(C(=O)Cn1cnnc1)C2 41356,C=CCCC(C(=O)NCc1ccnc(OC)n1)NC(c1cnc(OC)nc1)=O 41357,C1(CNC(CN(C)C)=O)CN(C(c2ncc3ccccn23)=O)CCC12CCOC2 41358,CC1(C)CC(NC(=O)C(N)=O)CCN(C(c2ccnc(F)c2O)=O)C1 41359,C1(C(=O)NC(C=C)C2CC2)CC2(CC(NC(=O)CC(C)(C)C#N)C2)C1 41360,C(=O)(C1CCCc2n[nH]cc21)NC(C)CNC(=O)CNC(=O)C(F)(F)F 41361,N1(C(C2N(C(C)=O)CCOC2)=O)CC(Nc2ncc3ccsc3n2)CC(C)(C)C1 41362,CC1(CCC(=O)NCC2CCC2NC(=O)CCCc2csc(=N)[nH]2)CCC(=O)N1 41363,CC1(OC(F)F)CCN(C(=O)COC(=O)NC2(C)CCCOC2)CC1 41364,c1(C(N2CCCC(n3cc(C(C)NC)nn3)C2)=O)cc(O)nc(Cl)c1 41365,C=CCC(CNC(C1CCSCC1)=O)NC(=O)C(C1CC1)SC 41366,C1(CNC(CN2C(C)CC2)=O)CN(C(=O)Cc2ccnc(C(F)(F)F)c2)CC1C 41367,C(=O)(N1CC(n2cc(CCCC(=O)N(C)C)nn2)CO1)C1C(C)(C(C)C)C1 41368,c1(C(=O)NC2CCN(C(c3ccc(COC)o3)=O)C2)cccc(CSC)c1C 41369,N1(CCNC(C2CCC(N(C(=O)CC3CCCC3O)C)C2)=O)CCC(C)(C)C1 41370,CC1(C)Cc2cccc(S(=O)(=O)NCCn3ccc(O)nc3=O)c2O1 41371,C1(O)(C(C)NC(=O)CCSc2nccn2C)CCN(C(=O)CCN(C)CCO)C1 41372,CN(CCCC(=O)NCC1(NC(=O)COC2CCCCC2)CCCC1)N=O 41373,c1(C(C(=O)NC(C)C(CO)NC(=O)C=CCN2CCCC2)O)ccccc1F 41374,N1(Cc2c3ccc(OC)cn3nc2)CCC(N=c2[nH]cnc3cc(I)sc23)C1 41375,c1(CN(C(C=CC(=O)NC(C2CCCC2)C)=O)C)ccccn1 41376,C(=O)(C1=CC2(CCOC2)C1)N1CCCC(C(=O)Nc2cncc(F)c2)CC1 41377,c1(C(N2CC(F)(C(=O)Nc3cnn(C4COC4)c3)C2)=O)ncccc1F 41378,C1(CC)C(NC(C2(F)CCC2)=O)CCN1C(=O)C(C)OCCOC 41379,c1(CC)cc(Cl)ccc1C(=O)NCC1(CNC(=O)C(C(C)C)NC)CCCC1 41380,C(c1ccc(OC)cc1OC)=CC(=O)NCC(CNC(C(COC)OC)=O)OC 41381,C(=O)(C(CC(C)C)N(C)C(c1cc(CO)on1)=O)N1CCC(C(CC)CC)C1 41382,Cc1cc(C(=O)NC2CN(C(=O)CC3CCCN3C)CC2F)c(O)nn1 41383,N1(C(C(C)OCC=C)=O)CC2CC(O)C1C2NC(c1cc(C)sn1)=O 41384,C1(CN)CCC(c2cn(C(C)C)nn2)CC1.C1(C(N)=O)(C(=O)CCC2CC2)CC1 41385,C12(CNC(CCOCC)=O)CCC(C1)N(C(c1ccc(C(F)F)nc1O)=O)C2 41386,N1(C(c2ccc(OC)c(O)c2)=O)CC2OCCN(C(=O)COC3CC3)C2C1 41387,c1(CC(N2CC(C(=O)Nc3n(C)nc(C)c3Cl)NCC2)=O)ccc2c(c1)CCO2 41388,c1(CCCCCC)ccc(C(N2CC3CC2C3C(=O)Nc2cncnc2)=O)cc1 41389,C1(C)(NC(C2C(NC(CCCNC(C)=O)=O)COC2)=O)C=CCCC1 41390,N1(C(CC(=O)NCC)=O)CCC=C(CNC(=O)C(C)CC2CCC2)C1 41391,N1(C(c2c(C)n[nH]c2)=O)CC2CCCCN2CC1CNC(c1cc(O)ncn1)=O 41392,C1(C(=O)NCC(C)NC(c2nccnc2N)=O)COc2ccc(Cl)cc2C1 41393,C1(CNC(CN(C(C)=O)C)=O)CCC(C)(C)CN1C(C1CCOC1)=O 41394,C(C)(C(=O)NC1COCCN(C(=O)Cc2ccc(Cl)cc2)C1)(C(C)C)OC 41395,N1(C(c2cc(C)ncc2)=O)CCN(C(=O)C(C2CCCCC2)O)C(CC2CC2)C1 41396,c1(N2CC(NC(=O)Nc3c(C(=O)OCC)nc[nH]3)C2)ncc2cc(Br)cnc2n1 41397,c1(C(C(=O)NC(C(CC=C)C)=O)N(C)C)c(F)cccc1F 41398,c1(CS(=O)(=O)NC(C(=O)N(C)C)(C)C)ccc(S(C)(=O)=O)cc1 41399,N1(C(CC(C(C)C)NC(C2CCSCC2)=O)=O)CC2(C1)CC(C)(O)C2 41400,CC(O)(C(=O)NC1CC(CC(=O)Nc2cc(C(F)(F)F)ccc2Cl)C1)C(F)(F)F 41401,N1(C(C2CC(OC)CN2C(C2(C3CC3)CC2)=O)=O)CC(OC)CC(O)C1 41402,C(=O)(CCS(=O)(=O)Cc1ccccn1)NC(=O)NC(c1cn(C(C)C)nc1)C 41403,c1(C(=O)NC2C(NC(C3(C(C)=O)CC3)=O)CCCC2)ccc(F)c(C#N)c1 41404,Cc1cc(N(C)CC2CCCCN2C(c2sccc2Cl)=O)ccc1[N+](=O)[O-] 41405,CC(C(C)C(=O)N1CCCC(NC(C23CCC(CC2)CO3)=O)C1)S(C)(=O)=O 41406,O=C1Nc2ccc(C(N3CCCC3C3CCCN3C(c3ccon3)=O)=O)cc2CO1 41407,C(CCN=c1[nH]c(N2CCOCC3(CCCCC3)C2)nc2ccccc12)N(C)C 41408,CN1CCN(C(C2CC2CF)=O)CC1CN1CCC(CC(=O)NCC2CC2)CC1 41409,c1(C(=O)NC2C(NC(c3n(OC)cnc3C)=O)COC2)cnc(O)n(C)c1=O 41410,c1(CCCC)cc(F)c(CC(=O)NCC2(N)CC(OCC)C2)cc1Br 41411,C1(CC(=O)NC(c2ccnn2C)C(=O)NCCc2cnc(C)o2)CCCNC1=O 41412,c1(C(N2CC3C(CNC(c4cn(CC)nn4)=O)(C3)C2)=O)ncc(F)cc1F 41413,N1(C(c2cnn(C)c2Cl)=O)CC2=C(C1)CN(C(=O)CP(C)(C)=O)C2 41414,C1(NC(c2c(C)nc(C)o2)=O)CCN(C(=O)Cc2cc[nH]n2)C12CCC2 41415,C1(COC)CC(C(C)(C)C)CN(C(=O)C(N2CCN(C(C)=O)CC2)=O)C1.C(C=O)O 41416,C1(NC(CC2CC(=C)C2)=O)CC2CCCC(C1)N2C(C1CCN(CC(C)C)C1)=O 41417,N1(C(c2c(C)cc(OC)c(OC)c2)=O)CCN(C(=O)C(F)(F)F)CC(C(=O)O)C1 41418,Cc1cc(CC(=O)NC(C)(C)CNC(C2CCCC(C)(C)O2)=O)ccc1O 41419,c1(OC)cc(F)ccc1CC(=O)N(C)CCN(C)C(c1nccnc1C(N)=O)=O 41420,c1(C(N2CCC(NC(C(C)c3ccsn3)=O)C2)=O)c(N)cc(F)cc1Cl 41421,C1(CC(=O)N(C)Cc2cn(CC(OCC)OCC)nn2)CCCCC1F 41422,c1(C(N2CC(CC)C(OC)CC2)=O)ccc2cnn(CCOC)c2c1 41423,C(=O)(C1CC(=O)Nc2ncccc21)N1CCCC(c2cc(C(C)CN(C)C)[nH]n2)C1 41424,N1(C(COC)=O)CCOC(C(N2CC(O)CC2C(C)C)=O)CC1 41425,N1(C(C(CC)n2nccc2C)=O)CCN(C(=O)C(C(C)(C)C)N(C)C)C2(CC2)C1 41426,c1(OC)cccc(Br)c1C(=O)NC12CC1CN(C(=O)C(=O)NCCC(N)=O)C2 41427,CC1C(=O)CCC(C(=O)N(C2CC2)Cc2ccc(F)c(Cl)c2)C1(C)C 41428,C=C1CC(CC(=O)NCC(C)(C2CC2)NC(=O)Cc2ccsn2)C1 41429,CC1=CCC(C(N2CCC(OCCNC(c3cc(C(N)=O)ccn3)=O)C2)=O)CC1 41430,C#CCCC(C(=O)NCC(O)CCC=C)NC(c1n[nH]c(=N)[nH]1)=O 41431,c1(C(=O)NC2C3CC(NC(C(=O)NCC)=O)CC32)ccc2c(c1)C(=O)CCN2 41432,c1(-c2onc(-c3nccc(N4CCC(OC)C4C)c3)n2)ccccc1I 41433,CCC(C)C(O)C(=O)N1CCCC1C1CCN(C(c2c[nH]ccc2=N)=O)CC1 41434,c1(NC(=O)NC(C)CC#N)ccccc1OCCNc1cccnc1 41435,c1(C(=O)NC(CNC(C(C)NC(C)=O)=O)(C)C)[nH]c2c(c1C)C(=O)CC(C)(C)C2 41436,CC(C)CC(C(=O)NCc1ccc(C(=O)NCC(=O)N(C)C)cc1)C(N)=O 41437,CCCC(C(=O)NCC1(NC(=O)C(C)NC(N)=O)CCCC1)OCC 41438,Cc1c(Cl)ccc(C(N2CCOCC2c2cn(C3CCCC=C3Br)nn2)=O)c1N 41439,N1(C(C2(C)CCCC2)=O)CCC2CCN(C(c3cccc(C(N)=O)n3)=O)C2C1 41440,CCCC(CNC(=O)Cn1cc(CNC2(C(N)=O)CC2)nn1)OCC 41441,C(=O)(CC(F)(F)C(F)F)NCc1nn(C)c(C(=O)NCCc2cocn2)c1 41442,C12(CNC(=O)C(O)c3ccsc3)CC(NC(C3CNC(=O)C3)=O)(C1)C2 41443,C1(NC(CCSCCC)=O)CC2CC1CN(C(c1ccnn(C)c1=O)=O)C2 41444,C1(CNC(c2c(C)c[nH]n2)C)CC2(CCC2)C(=O)O1 41445,c1(C(=O)NC2CN(C(C3(O)C(C)(C)C3)=O)CC(F)C2)cc(F)c(F)cc1F 41446,C1(NC(CCC)=O)CC2CCC1N(C(=O)COc1cccc(Br)c1F)C2 41447,C12(C(N3CC(=CC)C3)=O)CC(CN(C(C3CCC(C)=C(C)C3)=O)C1)C2 41448,CC(C)CC(C(=O)NC(c1cccnc1O)C)NC(C1CCCC1C1CC1)=O 41449,C(=O)(CC(O)CNC(=O)COC1CCC1)N(C1(C)CC1)CC 41450,CC1CC(C(N2CCC(C(=O)N(CCC(=O)N(C)C)C)CC2)=O)CCO1 41451,C1(CN(CCCNC(C(CC=CC)C)=O)Cc2cccnc2)CCC(C)=C(C)C1 41452,C12(C(=O)NCC(C(C)O)O)CCC(NC(=O)CC3CCCOC3)C1C2 41453,N1(C(C(C)=CC)=O)CCN(C(C2CC3CCC2O3)=O)C(c2ccc(F)c(F)c2)C1 41454,C=Cc1cnn(C)c1C(=O)NCC1CC(C)(C)CN1C(=O)CCc1cc(Cl)no1 41455,C1(NC(CN(C)C2CC2)=O)CCC(N(C)C(c2cnc(-c3ccsc3)s2)=O)C1 41456,c1(CCOC(C)C(=O)NC2(CNC(C3CS(=O)C3)=O)CC2)ccccc1 41457,S(=O)(=O)(c1ccc(NC2CCCCCC2)c(F)c1)NC(C1CC(O)C1)C 41458,C(=O)(C1=NOC2(CCCN(C(=O)C(O)Cc3cccc(Cl)c3)C2)C1)NCCOC 41459,Cc1cccc(C2CCCCN2C(CC2CC2(Cl)Cl)C(=O)NCCC#N)c1C 41460,C(=O)(C1CCc2ccc(Cl)nc21)NCC1(OC)CN(C(C(CCC)C)=O)C1 41461,c1(C(N2CC3C(NC(C4C(C)(C)CO4)=O)C3C2)=O)cccc2c1OC(C)(C)C2 41462,c1(OC)cc(Br)ccc1C(=O)N(CC(C)NC(c1cc(F)ccc1C)=O)C 41463,CCCCC(CNC(c1c(C2CC2)noc1C)=O)NC(=O)C(C1CC1)OCC 41464,Cc1cc(=NCCCOC(C)C)[nH]c(N2CCC3(CCC(C)C3)C2)n1 41465,c1(OC)cc(CC(=O)NCC2CN(C(C3CC3C(N)=O)=O)CC2C)ccc1C 41466,N12CCCCC1CNC1CC(C(C)C2=O)C1.c1(C2C(C(=O)NC)C2)ccccc1 41467,C#Cc1ccc(F)c(C(=O)NCC2CC(OC)CN2C(c2cnn(C)c2N)=O)c1 41468,CCC(CCOC)C(=O)NC1C=CCN(C(=O)CC(C)(F)F)C1 41469,C1(C(N2CCC(NC(CCc3nc(C)sc3)=O)C2C)=O)CCc2nc[nH]c2C1 41470,c1(CCN(CCCNC(=O)OC(C)(C)C)C(N)=O)ccccc1.C1(=O)C(=O)NN1 41471,N1(C(c2cc(C)c(F)nc2)=O)CCc2ccccc2C1CNC(=O)C1=COCC1 41472,C1(C(C)N(CCOC)C(=O)NC(C)(C)CCO)CCCCC1 41473,CC1(C)CCN(C(C2CSCC(=O)N2)=O)CC1CNC(c1snc(Cl)c1Cl)=O 41474,c1(C(=O)NCC(CNC(COCCCC)=O)O)c(-c2cccs2)nnn1C 41475,c1(C(=O)NCC(CC)(C)NC(=O)COCC2CCOC2)ccc(CO)c(Cl)c1 41476,N1(C(C(C)(c2cccs2)N(C)C)=O)CCC2(CCC(=O)NC2)C1 41477,Cc1ccc(F)c(C(=O)NC2CC(C)CN(C(=O)CC3CCCOCC3)C2)c1F 41478,C(=O)(C1OCCc2ccc(C)cc21)N1CC2N(C(COCC=C)=O)CC(C2)C1 41479,C1(CC)CCN(C(=O)C(CC)NC(c2ccc(CC3CCCCC3)o2)=O)CC1 41480,C#CC1(NC2CCn3nccc3C2)CC2(CCCC2)C1 41481,c1(NC(CCSCCCC)=O)cccc(NC(c2cc(Br)sn2)=O)c1 41482,Cc1ncc2n1CCN(C(C1CCCC1CNC(C1(C3CC3)CC(=O)C1)=O)=O)C2 41483,C(=O)(CC(C)(C)CC(F)F)N1CC(NC(Cc2c(C)cc(C)nc2O)=O)C(F)C1 41484,C1(C(=O)NCC2N(C(c3c(C)nc(C4CC4)o3)=O)CC(O)C2)CCN(C)S1(=O)=O 41485,N1(C(C(=O)NCC(F)F)=O)CCCC(C2CC2NC(c2ccccc2O)=O)C1 41486,CN1CC=C(CC(=O)N2CCC(O)(CNC(C3Cc4ccncc4C3)=O)C2)CC1 41487,C12(C(=O)NCC3NC(=O)OC3)CC1CCN2C(c1cnn[nH]1)=O 41488,N1(C(c2cnn(C(CC)C)c2C2CC2)=O)CCN(C(C2CC23CCC3)=O)CC1C 41489,C(CCCCC(C)C)NC(N(CC)CC1CCCCN1C(C)=O)=O 41490,Cc1cc(C)c(C(=O)NCC2(C(C)NC(c3cocc3C)=O)CC2)c(O)n1 41491,C1(NC(CC)=O)CC2CCC(C1C)N2C(c1cnn(C)c1C(F)F)=O 41492,C1(C(N2C(CNC(c3c(C(C)C)ocn3)=O)CCC2)=O)CCC(C#N)CC1 41493,Cc1ccc(F)c(CC(N2CC(CNC(c3nnsc3C)=O)C3(CC3)C2)=O)c1 41494,N1(C(=O)OC(C)(C)C)CCC(n2cc(CCNC(C(N)=O)c3ccc[nH]3)nn2)C1 41495,C1(OC(c2ccc(OCC)c(F)c2CC)=O)CC2(CCOCC2)CCO1 41496,CC(N=[N+]=[N-])C(=O)NCC(C1CC1)NC(=O)CC1COCCOC1 41497,CCCCCCC(CC)C(=O)N1CC(NC(=O)C(C)(C)F)C(O)C1 41498,C1(CC(=O)NCCC(C)NC(c2cscc2C(F)F)=O)COC(C)(C)C1 41499,CCC(CNC(c1cn(C)nc1OC)=O)(CC)NC(=O)C(C)C(=O)OC 41500,N1(C(C(CC)c2ccccc2)=O)CCCC2(CCCCN2CC2CCOC2C)C1 41501,Cc1ncc(C(=O)NOC(CC(C)C)C(=O)NCCN(C2CCCC2)C)c(=N)[nH]1 41502,C12(CNC(C3(C)CC3)=O)CC1CN(C(=O)CCCCc1cnn[nH]1)C2 41503,c1(C(N2C(C(N3CCC=C(F)C3)=O)CCC2)=O)cccc2cc[nH]c12 41504,C1(CNC(C2(CCCC)CCCC2)=O)CC(OC)CN1C(=O)Cc1cccs1 41505,c1(NC(C(=O)NC2(C)C(C)C2)=O)cccc(NC(=O)C(F)(F)F)c1 41506,N1(C(C(CC#C)O)=O)CC2CCC(CNC(=O)Cc3nc(C4CC4)cs3)(C2)C1 41507,C1(NC(CC(CN(C)C)O)=O)CN(C(=O)COCc2ccncc2)CC12CCC2 41508,CC1C(C(=O)N2CCC(C)(C)C2C(=O)NC2CC(C(C)(C)C)C2)=NOC1C 41509,C1(C(=O)NC(CCCNC(C(CC)n2ccnc2)=O)C)CC12CCCCCC2 41510,CCC(CC)C(=O)NCCC1(COCCC(=O)Nc2ccccc2C(C)C)CC1 41511,c1(C(C)NCCO)cccc(NC(C(=O)NC(C)C)=O)c1.S(C)(=O)(=O)N 41512,Cc1cc(N)c(C(=O)NCC(C)(C)OCCNC(=O)CN2CCC(C)C2)nc1C 41513,C(=O)(CC(CCCC(C)C)NC(C1(NC)CC2(C1)CC1(CC(F)(F)C1)C2)=O)OCC 41514,CC1(NC(=O)CC(C2CC2)NC(=O)CCc2cncnc2)CCCOC1 41515,N1(C(CC2C(C)CCO2)=O)CCC(NC(c2cccn(C)c2=O)=O)C(CO)CC1 41516,c1(CCC)nc(C)c(C(=O)NCC2CC(NC(C3CCOC3(C)C)=O)C2)o1 41517,CCCCC(C)C(=O)N1CCC(CCC(=O)Nc2ccc(Cl)cc2O)C1 41518,N1(CC)CCN(C(C23CC(CO)(CN2C(C2(C)CC(C)=NO2)=O)C3)=O)C(C)C1 41519,N1(C(C=CCC)=O)CC(C)N(C(c2cc(CC(C)C)c[nH]2)=O)CC1C 41520,C1(C(=O)OCC)CN(C(=O)CC2COCCN2CC(F)(F)F)C2(CCC2)CO1 41521,N1(C(c2c(C)cccc2)=O)CCC2COC(CC(=O)Nc3cccnc3)C2C1 41522,N1(C(C2C(COC)CC2)=O)CCCC1C=CC(=O)NC1(CO)CCC1 41523,C(=O)(C(O)CC(C)(C)C)NC1C(C)N(C(c2cnc(O)s2)=O)CCC1 41524,N1(C(c2ccc(C(C)=O)s2)=O)CC2CC(NC(c3oncc3C)=O)CC1C2 41525,c1(CC)ccc(NC(=O)CCOCCCNC(=O)CCOC)c(C)n1 41526,C(=O)(C(C)(O)Cn1ccccc1=O)NC1C(NC(c2ccc(OC)s2)=O)C1 41527,C=C(Br)CC(C)(C)C(=O)N(C)CCN(C(c1noc(C2CC2)c1C)=O)C(C)C 41528,C1(O)(CNC(C2C(=C)C2)=O)CCN(C(=O)CC2COC(=O)C2)CC1 41529,C1(C(=O)NCC(CC)(C)OC)C=CCN(C(C2CC2Cl)=O)C1 41530,C(=O)(C(C)N(C)C(C1CC(=O)C1)=O)NCCN(CCC)CCC 41531,n1(C2CCC(C(C)C3CC3)C2)cnc2c(N3CCC(S(N)(=O)=O)CC3)ncnc12 41532,Cn1cc(NC(c2nnnn2-c2ccccc2)C=CC2CCCC2)c(C#N)n1 41533,c1(C(=O)NCC2COCCN2C(=O)C(O)C2CC2)nc[nH]c2nccc1-2 41534,C1(OC)COc2c(C(=O)OC(c3ccccc3Br)C(=O)O)cnn2C1 41535,C1(C(N2C(C(=O)O)CC(CC)C2)C)CC2CC(=O)C1C2 41536,C1(C(=O)NCc2snnc2C2CC2)CSCCN1C(=O)CCCCC1CC1 41537,CC1CC(NC(=O)COc2ccccc2)CN1C(c1ccsc1Cl)=O 41538,c1(C(=O)NCC(CN(C(c2cnc(C)n2C)=O)C)(C)C)cnc2ccc(F)cn12 41539,c1(N2CCC(Cc3c(Br)cc(C)c(Cl)n3)CC2)cc(Cl)cc(Cl)c1[N+](=O)[O-] 41540,C(=O)(CCCCN1CCCC1)N(CCCCNC(CCOCC#C)=O)C(C)C 41541,CC1=CCC(C(N2CC(CO)(NC(=O)CC(O)CN(C)C)C2)=O)CC1 41542,c1(CN(CC(C)(C)[N+](=O)[O-])C(=O)C(=O)NC2(O)CCNCC2)c(Br)cncc1Br 41543,c1(CNC(C2C(OC(C)=O)C2)=O)ccnc(C(=O)NCCC2CCOC(C)C2)c1 41544,C(C)(CN=c1ccnc(NCc2nnc(O)n2C)[nH]1)(C1CC1)OC 41545,Cn1ccc(=NC(=O)C2CC(O)CN2C(c2ccn(C(C)(C)C)n2)=O)[nH]1 41546,C1(C(=O)NC(C(=O)NCC(CSC)(C)O)CCF)C2CCC(C2)C1C 41547,c1(OC)ccc(F)c(F)c1CN1CCN(Cc2cc(C(F)(F)F)nn2C)CC1C 41548,C(=O)(CCCCC(N)=O)NCC(C)CNC(c1cnc(OC(C)(C)C)nc1)=O 41549,Cn1cc(C(N2CCC3(CC(NC(=O)OC(C)(C)C)C3)C2)=O)c(=O)[nH]c1=O 41550,c1(CC)nnc2n1CCCC2C(=O)NCC1(NC(=O)C(C)C(F)F)CC1 41551,C(=O)(C(C)(O)COC)N(C)CC1N(C(CC(=O)NC)=O)CCC1 41552,CCCCC(O)CCC(=O)NCC(C)(C1CC1)NC(C1CCCCN1N=O)=O 41553,C1(C)(C(=O)NC(C)CCN(C(=O)Cc2nccn2C)C)CC2CCC(C1)S2 41554,Cc1cc(NC2(c3nnnn3C3CCC3)CCOCC2F)cc(F)c1Br 41555,C(=O)(CC1=CCN(C)CC1)N1C(CNC(C2(C(=O)OCC)CCC2)=O)COCC1 41556,C1(C#N)(C(=O)NCCCOCCCNC(c2ccc(CC)cn2)=O)CCCCC1 41557,c1(NC(N2CCOC(c3cn(CC(F)(F)C(F)F)nn3)C2)=O)ncc(Br)cc1F 41558,C12(CNC(COCCOC)=O)CC(CO1)N(C(c1cnn(C)c1SC)=O)C2 41559,C1(CC(=O)NCC2OCCN(C(c3c(C)cn(C)c3)=O)C2)COCC(C)(C)O1 41560,CCCC(CCC)C(=O)NCC(C)NC(C1CC=C(C(C)C)CC1)=O 41561,N1(C(C2(C)CCC2)=O)CC2CS(=O)(=O)CC2(CNC(c2c(F)cccc2F)=O)C1 41562,C1(O)(C(N2CCCC(NC(=O)CCC(F)(F)F)CC2)=O)Cc2ccccc2C1 41563,CCC(CC(=O)OC)NC(C1(N(C)C)CCCSC1)=O 41564,C1(CNC(CC2CC(OC)C2)=O)(CO)CCN(C(c2cc(C)cc(C)n2)=O)CC1 41565,c1(NC(C2(C)CCCC2)c2nnnn2CC(F)F)ccc(CCF)cc1 41566,c1(SC)ccsc1C(=O)NCCN(C(=O)C(C)SC1CCOCC1)C 41567,c12cccc(c1)C(c1n(CCCOC)nnn1)N2.O(C(F)F)CC 41568,C=CC1CCCCN1C(C12CC1CN(C(=O)CC(C)(C)Cc1ccccc1)C2)=O 41569,c1(CNC2(C(=O)NC3(C(=O)NCC)CCCC3)CC2)ccc(-n2cccn2)cc1 41570,c1(C(N2CCC(CCNC(C(C)CO)=O)CC2)=O)cccc2c1CC(=O)N2C 41571,C12(CNC(c3cnc(Cl)s3)=O)CCCCC1N(C(=O)CC1CC(F)C1)CCC2 41572,c1(C(=O)NC2C(NC(Cc3c(C)ccs3)=O)CC2)cnn(C(C)(C)C)c1C 41573,n1(CCOC)cc(C(=O)NCC2COC(CNC(c3nn[nH]c3Cl)=O)C2)c(C)n1 41574,S(=O)(=O)(c1c(Cl)ccc(C)c1F)NC(C(=O)OCC)(C)Cc1ccccc1F 41575,CC1(F)CC2(CN(C(C3(C)CCN(C(c4cc5n(n4)CCO5)=O)C3)=O)C2)C1 41576,C1(C(=O)NCC(CN(C(=O)CCc2ccccn2)C)O)CC(=O)CCO1 41577,CCC(CC(=O)NCC(CC)(CC)NC(c1ccc(CC(N)=O)cc1)=O)C1CC1 41578,CC1CC(C(=O)N(C)CCNC(C2(CF)CC(F)(F)C2)=O)CCO1 41579,C#CCC(C)C(=O)NCC(C)(C)CN(C(=O)C(c1ccccc1)F)CC 41580,C1(CNC(CC2ON=C(C)C2)=O)CCC(NC(C2CCN(C)C2)=O)CC1 41581,CC(CCCc1cn(C(C)C(=O)O)nn1)C(=O)NC1CCN(C2CCCCC2)C1 41582,CCC(C(=O)NC1CCN(C(c2oc(C)nc2C)=O)CC1O)C(F)(F)F 41583,CC1(C)CCN(CCNC(=O)C(c2ccoc2)NC(=O)CSC2CC2)C1 41584,c1(CN(C)C(N2CC(C(O)CO)C2)=O)cc2c(s1)CCC(C)(C)C2 41585,c1(C(=O)NCCCC(C)NC(c2cncc(SCC)n2)=O)ccc(N)c(C)c1 41586,Cc1ccc(F)cc1C(N1CC(CNC(c2nc(C3CC3)cs2)=O)C(O)C1)=O 41587,N1(C(Cc2c(C)nc(CC)s2)=O)CC(CC(=O)OC)C(C2CC2)C1 41588,c1(CC)nnc2c(C(N3CCC(NC(C4(O)CC4)=O)CC3C)=O)cccn12 41589,C(=O)(C(C)(C)C(C)O)NCCC1(OC)CN(C(=O)Cc2c(Cl)c(CC)nn2C)C1 41590,c1(N(C)C)ncnc(N2CCOC(CNC(C3(O)CCOC3)=O)C2)c1[N+](=O)[O-] 41591,C1(CC)(NC(=O)CN2CCOCC2=O)CCCN(C(=O)C(CC)n2ccnc2)C1 41592,N1(C(c2ccc(F)c(C#N)n2)Cc2n(C)nnn2)Cc2ccccc2OC2(CCOC2)C1 41593,C(=O)(CCCCC1CC1)NCC(C=C)O.C12(CC1)C(=O)N2 41594,c1(C(N2CC3CN(C(c4ccon4)=O)CC32)=O)cn2cccc(Br)c2n1 41595,C12(CNC(c3ccc(N)cn3)=O)CCC(NC(C3CCCC(=O)N3)=O)(CO1)C2 41596,n1(C(C)C)cc(C(=O)NC2CC(O)CN(C(c3cn(C)[nH]c3=N)=O)C2)ccc1=O 41597,N1(C(COC2CCCC(C)C2)=O)CC2CC(C1)C2NC(c1ccnc(O)c1)=O 41598,c1(C(=O)NCC2CCC(CNC(C3CCC(C)(CC)O3)=O)C2)ccc(C)c(O)c1 41599,CCC(C)C(=O)C(=O)NC1(C(=O)N(C(C)CC(C)C)C)CC(O)C1 41600,N1(C(C2(C)C=CCC2)=O)CCCCCC(NC(=O)C(c2ccc(O)cc2)=O)C1 41601,N1(C(C(C)CBr)=O)CCC2(CCN(C(c3cc(C4CC4)nn3C)=O)C2)C1 41602,c1(OCC=C)c(C(=O)OC(CC(=O)NCC(C)NC(=O)COCC)=O)cccc1C 41603,CC12CC(NC(=O)CC3CC4CC4C3)(C1)C1(CCN(C(c3nncs3)=O)CC1)O2 41604,N1(C(c2c(Cl)ccc(OC)c2)=O)CC2CCC1C(CNC(C1CCOCC1)=O)C2 41605,c1(C(N2CCC(N(C(C(CC)O)=O)CC)C2)=O)cc(F)c(Cl)c([N+](=O)[O-])c1 41606,c1(-c2cc(C(=O)NCC(C)N(C(C(C)=C(CC)C)=O)CC)no2)ccc(Cl)cc1 41607,CC1(CNC(C2CCOC(=O)N2)=O)CCCN(C(c2cn(CCO)nn2)=O)C1 41608,c1(CC(N2C(C(N3CCCOCC3)=O)CC(=C)C2)=O)cccc(Cl)c1F 41609,CC1(CNC(c2ncn3c2CCC3)=O)CN(C(c2cccc(Cl)c2)=O)CCO1 41610,C1CCCC(N=c2[nH]c(=NCC3CCSC3)c3ccccc3[nH]2)C1 41611,c1(C2C(C)C2)ccc(NC2(CNC(=O)OC(C)(C)C)CCCCCC2)c(F)c1 41612,N1(C(C=C(C)c2cccs2)=O)CCCC1C1CCCN1C(=O)CCCN=[N+]=[N-] 41613,c1(C(C(=O)NC(C)C)N(CCOC)C(C)C2CC2)csc(Cl)c1 41614,N1(CC(N2C(CCC)CCC2)=O)CCN(C(C2(SC)CCC2)=O)CC1 41615,C(c1ccc(C(=O)NC(C)CNC(=O)CC(C)C2CC2)cc1)=CC(=O)OC 41616,C1(C(N(C)Cc2ccsc2)=O)CCN(C(=O)CCOC2CCC2)O1 41617,Cc1[nH]c(C)c(C(=O)NC2CC(C)(NC(c3ccnn3CCF)=O)C2)c1C 41618,CN1CC(NC(c2occc2CNC(C2C3CCCC23)=O)=O)C(F)(F)C1 41619,C12(C(N3CC(C)C(NC(C4(F)CCCCC4)=O)CC3)=O)C3CC(CC13)C2(F)F 41620,N(C(=NCCOc1ccc(Cl)cn1)NCC1CCC(F)CC1)C(COC)C 41621,N1(C(c2cnn(C(C)C)c2Br)=O)CC2(C1)CN(C(=O)CC#N)C2 41622,C1(N(CC(=O)NCCN2CCN(C(C(C)(C)C)=O)CC2)C)CN2CCC1CC2 41623,c1(C(=O)NC2CCC(CCC(=O)NCCOCC=C)C2)nc(C)ccc1C 41624,C1(NC(=O)COc2cccnc2)CN(C(=O)CCc2ccc(Cl)cc2)CC1F 41625,C1(C(=O)NCC23CC(CO)(CO2)C3)(OC)CCN(C(c2cncc(CO)c2)=O)C1 41626,C1(C#N)(C(=O)NCCc2c(C(=O)NCC3(O)CCN(C)C3)c[nH]n2)CCOCC1 41627,c1(CC(=O)Nc2cccc(NC(=O)CC3CCCNC3=O)c2)cc(Cl)ccc1Cl 41628,c1(C(N)=O)cc(CC(=O)NCC2(O)CN(C(C3(n4nccn4)CC3)=O)C2)on1 41629,c1(CC)c(C(=O)NCCCC2CCCN2C(C2CC2C(F)(F)F)=O)cccc1C 41630,CCCC(C)CC(=O)NCC1CCCN(C(c2cc(CC)ccc2C)=O)C1 41631,CCCC(C)CN=c1cccc(S(=O)(=O)NCCCn2ccnc2CC)[nH]1 41632,c1(OC)ccc(C)c(OC)c1C(=O)NCC(C)CNC(=O)CCC1CC(OC)C1 41633,C12(C(=O)OC)CCN(N3CC(c4cccc5[nH]ccc45)C3)CC1C2 41634,C1(C(N(CC(=O)NCCC2CC=CCC2)CC)=O)C(C(C)=O)C1(C)C 41635,c1(CC)[nH]nc(C(=O)N(CCCN(C)C)CCNC(=O)C(O)CC2CC2)c1Cl 41636,C=CCC(C)C(=O)NC1CC(N(C(=O)Cc2sccc2-c2ccccc2)C)C1 41637,N1(C(C(CC)N(C)C)=O)CCC2(C=C(C(=O)N3CCCN(C)CC3)C2)C1 41638,c1(C(N2C(CNC(c3ccc(Br)nc3Br)=O)COCC2)=O)cc2cccnn2n1 41639,C(=O)(C(CC(C)C)NC1(CCF)CC1)N(CC(COC)O)C 41640,C1(O)(CCNC(C(CC)C#N)=O)CCCN(C(=O)COc2cc(Cl)ccc2C)C1 41641,N1(C(C2C(=C)C2)=O)CC2CCC1CN2C(C1CC(c2ccccc2)(OC)C1)=O 41642,c1(C(=O)NC2CC(F)(CNC(C3CC(C)OC3)=O)C2)ccc(-n2cncn2)c(N)c1 41643,N1(C(C(CC)=CC)=O)CCCC12CCN(C(C1CCN(C3CC3)C1=O)=O)C2 41644,CN1N=C(CC(=O)N2CCC=C(CNC(=O)C(C)(C)C3CCCO3)C2)CC1=O 41645,N1(C(C2(CC)CC2(F)F)=O)CCC(CF)(NC(c2ncoc2C)=O)C1 41646,N1(CCOC)CCN(C(=O)Cn2cc(CCC3(OC)CCC3)nn2)CC1 41647,CCCCCCC(F)C(=O)N(C1(C)CCN(CCOc2c(C)cccc2C)C1)C 41648,C(CN=C(NCCn1ncc(Br)n1)N(C)CC1CCOC1)SC(C)(C)C.CCO 41649,c1(OC)c(NC(C2(NC(=O)OC(C)(C)C)CC3CCC2C3)=O)c(C)nn1C 41650,c1(NC(C)C(=O)OCC(C)CNCCCC)c([N+](=O)[O-])c(C)nn1CC 41651,CC1(C)CCCC(CC(N2CC(CNC(c3cncc(N)c3)=O)C2)=O)O1 41652,CC1CC(N(C(=O)COC2CCN(C(C3(C)CCCCCC3)=O)C2)C)CC(C)C1 41653,C(CO)(CC(C)(C)C)NC(C(CC=C)NC(=O)Cc1ccc(F)nc1)=O 41654,CC1CN(C(c2cscn2)=O)CC1CNC(c1cnn(CC(F)F)c1)=O 41655,c1(C2N(CC)CC2)nc(-c2ccc(OC(C)(C)C)cc2)nn1CCCN(C)C 41656,Cn1c(C(=O)NC2CN(C(=O)CCC3CCCCO3)CCC2F)cc(Cl)c1Cl 41657,N1(C(C(C)CC2CCC2)=O)CCOCC(C(=O)NC2CN(C)CC2(F)F)C1 41658,c1(OC)ccc(C(C(=O)Nc2ccccc2Cl)OCCOC)c(NC(=O)NC)c1 41659,CC(C)CC(O)C(C)C(=O)N1CSCC1C(N1CCCC(C)C1CO)=O 41660,C1(C(N2CCN(CCCNC(=O)CCOCC(F)F)CC2)=O)C2CCCCCC12 41661,N1(C(Cc2nn(C)c(Cl)c2)=O)CCC2CN(C(=O)C(O)CC3CC3)CC12 41662,Cn1ncnc1C(N1CCCC1C(=O)NCc1ccccc1)C(=O)NC1CCC1 41663,CC#CCC(C(=O)NCC(C)(C)C1(O)CCC1)NC(C1CN2CCC1C2)=O 41664,N1(C(CCCCC)=O)CC2(C1)SCCC2NC(c1ccccc1OC)=O 41665,c1(SC)nc(N(c2ccc(N3CCCCC3)cc2)C)nc(N)n1 41666,c1(C(=O)NC(c2c(C(=O)NCCCC=CC)con2)C)cc(CC)oc1C 41667,N1(C(COCc2cc(C)no2)=O)CC(NC(c2ccc(=O)oc2)=O)C(O)C1 41668,C1(O)(C(N)=O)CCCN(C(c2ccc(CNC(=O)CC3CCNC3=O)cn2)=O)C1 41669,C1(NC(C=COCC)=O)CS(=O)(=O)CC1NC(c1cc(Br)sn1)=O 41670,C1(NC(CCN(C)CC)=O)CCN(C(=O)CC2CC23CC3)C1C 41671,C(CN=c1nc(CC2CC2)[nH]s1)CC1CCCN(C(c2cnc(OC)s2)=O)C1 41672,C1(N(C(=O)COc2cn[nH]c2)C)CCCCN(C(=O)C=Cc2cccc(O)c2)C1 41673,c1(NC(=O)OC)cccc(CNC(=O)CN2CCC(C)CC2)n1 41674,N1(C(C(CC(=C)C)OC)=O)CCC2CN(C(=O)C(N3C(=O)CCC3=O)C)C(C)C12 41675,CCC(C)(CNC(=O)CCc1ccccc1F)C(N)=O 41676,c1(COC)nn(C)cc1C(=O)NCC(C)(CO)NC(=O)Cc1cncc(O)c1 41677,C1(C(=O)NC2(CCCC(=O)NCC3C(CO)C3(F)F)CCC2)CC2C=CC1O2 41678,C(=O)(C(C(=O)NCC1CCN1C(c1cc(O)n(CC)n1)=O)C(C)C)OCC 41679,C(=O)(CC(C)C(C)(C)CC)NCCCOCCN(C(CCC=CC)=O)C 41680,Cn1c(C(N2C3CN(C(=O)Cc4cccnc4Cl)CC23)=O)cc2ccccc12 41681,Cc1ccc2oc(C(=O)NC3C4CCN(C(C5(C)CCCOCC5)=O)C34)cc2n1 41682,c1(C(=O)NCc2nc(CNC(c3ccc(C)s3)=O)sc2)ccn2nncc2c1 41683,c1(CC(=O)NCC(CN(C(C(C)SC)=O)C)C)cncc(C)c1 41684,c1(C(N2CC(C(C)NC(C3CCCCC3C)=O)C2)=O)cn(C)c2ccccc12 41685,C1(F)(CNC(C2N(CCC)CCC2)=O)CCN(C(c2nc(O)c(C)s2)=O)C1 41686,CC(=O)CCCC(=O)N1CCC(CCC(=O)NC2C3CCCCCC23)C1 41687,C(=O)(C(F)(F)CCC=C)N(C1CNC(=O)C(C)O1)C.C1(CO)CC1 41688,CC(C(=O)N(C)Cc1cnn(-c2ccccc2)c1)N1C(=O)COc2ccccc21 41689,Cc1cccc(SC(C)CC(F)(F)F)c1.c1(C2Cn3nnnc3S2)ccccc1F 41690,CC(C)(C)CC(O)C(=O)NC(Cc1cc[nH]n1)C(N1CCCCCC1)=O 41691,c1(C(=O)NCC(CN(C(C(C)OC)=O)C)C)cn(-c2ccc(F)cc2)nc1C 41692,CCC(CC(=O)N(CCC(C)NC(=O)COC1(C(F)(F)F)COC1)C)OC 41693,c1(CNCC2N(C(c3nc(CC)oc3)=O)CCCC2)n[nH]c2ccccc12 41694,C1(C)(C(N(CCNC(=O)C=C(C)C)CC)=O)CCC(=O)NC1 41695,N1(C(C(C)OCC#C)=O)CC(NC(c2sccc2OCC)=O)C2CCCCC12 41696,C1(CCOC)(NC(=O)C=CC2CCCN2C)CCN(C(=O)C(C)(C)C2CCC2)C1 41697,C(=O)(CC(C)(F)F)N(CC(C)O)CCNC(C1C(C)C1C)=O 41698,C=CCCCC(C(=O)N1CCC(n2ccnn2)C1)NC(c1cn(C)cn1)=O 41699,N1(C(C2CC(C#N)C2)=O)CCC2(NC(c3ncccc3Cl)=O)CCCC12 41700,c1(NC(C(CC=CC)NC(=O)Cc2ncoc2C)=O)cc(C)ccc1CO 41701,c1(C(N2CC3C(C(N4CC(C#N)(COC)C4)=O)C3C2)=O)cccc2ccnn12 41702,CCC(C)CCNC(C1CCN1C(=O)COCCCOC)=O 41703,N1(C(C(CC)Cl)=O)CC(NC(C2CC(O)CN2)=O)C2(COC2)C1 41704,n1(CC(=O)NC2CCCC(NC(Cc3c(C)nc[nH]3)=O)C2)cc2ccccc2n1 41705,C(=O)(C(CC)CC(C)C)NCCCC(C)NC(c1c(CC)c(F)ccc1)=O 41706,C1(C(C)NC(C(C)OCCC=C)=O)CCCN(Cc2cc(OC)ns2)C1 41707,N1(C(c2c(C)cccc2F)=O)C2CCC1CN(C(C1CCC3(CC1)CC3)=O)C2 41708,Cc1nn(C)c(Cl)c1CNCCC(N1CCOCC(C(=O)NC(C)(C)C)C1)=O 41709,CCC(C(=O)N1CCC(C(=O)NC(c2nccn2CC)C)C1)C(C)(C)CC 41710,c1(C(=O)NC(CC)CNC(c2ncccc2Cl)=O)cc(Cl)sc1S(N)(=O)=O 41711,c1(C(=O)NCCC(CC)(CC)NC(=O)CCCOC(C)=O)nccc2nn[nH]c12 41712,Cc1nc(CNC(C2CCN(c3cc(-n4cncn4)ncn3)CC2)=O)sc1C 41713,CCN=C(NCC1CCN(c2ccc(COC)cn2)C1)NCCc1ccccc1Cl 41714,CC(O)(C(=O)NCCCCNC(C12CC(c3ccccc3)C1C2)=O)C1CCC1 41715,C1(NC(Cc2c(OC)cccc2)=O)CCSC12CN(C(C1CCCOC1)=O)C2 41716,C1(OCC)COCCC1CC(=O)NCC(=C1CN(C(c2nccs2)=O)C1)F 41717,CCCCC(Cc1cn(C(=O)NNC(=O)CCOC)nn1)CCC 41718,CC(C)CC(CNC(C1COC(=O)O1)=O)NC(=O)CSc1ccccc1 41719,C12(CNC(c3c(OC)nsc3)=O)CCC1CN(C(C1CC(O)CN1C)=O)C2 41720,CS(=O)(=O)C1CCCN(C(=O)CC2CCN(C(=O)CCc3ccco3)C2)C1 41721,N1(C(COCCCC#C)=O)CCCC(O)(CCNC(c2c(Cl)csc2Cl)=O)C1 41722,Cc1c[nH]c2ncnc(N3CCSCC3C(=O)NC(c3cccc(Cl)c3)C)c12 41723,c1(NC(C(c2c(C)nccc2)C)=O)ncc2c(n1)COCC2 41724,C(=O)(C(C)(C)C(N)=O)NCCCC(C)NC(=O)C(C(C)(C)C)N1C(=O)CCC1=O 41725,N1(C(C=C(CC)CC)=O)CCC(O)(CN(C(=O)Cc2cnn(C)c2)C)C1 41726,O=C(CCCCCCCO)NCCCN(CCO)C(C1CC(=O)N(C(C)(C)C)C1)=O 41727,c1(C(=O)NC2CCN(C(C3COCC4(CCC4)O3)=O)C2)cc2cc(F)ccc2s1 41728,CC1(C(=O)Nc2cscn2)CCCN1C(c1nc(Cl)sc1Cl)=O 41729,CC1CCCC=C1C(=O)N(C(C)CNC(c1cc2ncccc2[nH]1)=O)C 41730,C(=O)(CCCC(C)(F)F)NCCC1OCCN(C(c2c(C)csc2)=O)C1 41731,C1(NC(C(Cn2ccnn2)NC(C2C=CCC2)=O)=O)CC2CCCC2C1 41732,N1(C(CNS(C)(=O)=O)=O)CCOC2CN(C(c3ccsc3C(F)F)=O)CC12 41733,C1(CC(=O)NCc2cc(C)on2)COCCN1C(C1CC1C(N)=O)=O 41734,Cc1ncc2n1CC(C(=O)NCCN(C)C(C1CC3(CCCC3)CO1)=O)CC2 41735,N1(C(COC)=O)CC(C)(C)CC1CNC(=O)C(O)C(Cc1ccccc1)OC 41736,N1(C(CC2CCN(C(c3c(C)c(Br)no3)=O)C2)=O)CCC2(CC1)CC(C)NC2=O 41737,N1(C(CC=CC=C)=O)CC(O)(CN(C)C(C2CC3CCC23)=O)C1 41738,N1(C(c2cn(C)nn2)C(=O)NC2CCCC2)CCCC(CN2CCCCCC2)C1 41739,N1(C(C(CC)N(C)C)=O)C2CCC1CN(C(=O)C(C)Oc1ccccn1)C2 41740,CC(C)CCC(C)C(=O)NCC1(CC(=O)OC(C)(C)C)CC1(F)F 41741,C1(CNC(c2ccc(OCC=C)cc2)=O)CN(C(=O)CC2(O)CC2)CCC1CO 41742,C1(NC(C(C=C)O)=O)CCN(C(=O)CN(C)C(=O)OC(C)(C)C)C12CC2 41743,C(=O)(C(C)(CC)OC)NCCN(C(c1cncc(C(F)F)c1)=O)CC 41744,N1(CC(C)C)CCC(C2CCCN(C(c3nccc4ccsc34)=O)C2)C1 41745,c1(CCNC(C2C=CCN2C(c2ccnnc2)=O)=O)ccc(F)cc1 41746,c1(C(N2CC3C(CNC(c4cnc(CCC)s4)=O)C3C2)=O)cc2nc[nH]c2cn1 41747,C1(COC)OC(c2nc(Cc3ccoc3)no2)CC1C 41748,C1(CC)CN(C(C2COCCOC2)=O)CCN1C(C12CCCC1(C(N)=O)C2)=O 41749,c1(C(=O)NCC(CNC(C(CCCC)N(C)C)=O)F)oc2ccccc2c1CO 41750,c1(C(=O)NCC(CC=C)NC(c2cccnc2)=O)ccc(Cl)c(OC)c1F 41751,C1(C(=O)NCC2(C)CCN(C(c3c(C)c(C4CC4)on3)=O)C2)CCCCNC1=O 41752,c1(C(=O)NC2(CNC(C(CC)CC3CCCC3)=O)CCC2)cc2cccnn2n1 41753,N1(C(C2(C=C)CC2)=O)CCN(C(c2cnc(Cc3ccc(Cl)cc3)s2)=O)CC1C 41754,N1(C(CC(C)F)=O)CC2CCOC2(CNC(c2cc(=O)cc(Cl)[nH]2)=O)C1 41755,C1(NC(=O)C2=CCCC2)CC2CN(C(c3nscc3Br)=O)CC2C1 41756,c1(-c2c(C(CC(N3CCCC3)=O)=O)c[nH]c2)ccc(-c2ccncn2)cc1 41757,CN1CCC(F)(C(=O)NCCCCCCNC(c2cccc(O)n2)=O)CC1 41758,CCC(C)(CNC(C1(F)CCN(C(c2ccc(CO)cn2)=O)C1)=O)C(N)=O 41759,C(=O)(C(C)C(CC)CC)N1CCCC(n2cc(C(C3CC3)OC)nn2)C1 41760,c1(C(C)(C)C(N)=O)ccc(NC(C2CC2c2cncc(Br)c2)=O)cc1 41761,C(=O)(C1=CC(O)C(O)C(O)C1)N1C(C(N2CCC(OC)C2)=O)CC1 41762,C(=O)(CC(F)(F)CS(C)(=O)=O)N1CCC(O)(C(C)NC(c2c(C)nccn2)=O)C1 41763,C(CCC(=O)NC(C)(C)CNC(c1nocc1C1CC1)=O)OCC=C 41764,c1(OC)ccnc(C(C(=O)NC2CCOC2)N(C2CCCCC2C)C)c1C 41765,N1(C(C2N(CC)CCC2)=O)CCC(C(=O)NC(CC2CC2)C(=O)NC)C1(C)C 41766,c1(OC)cc(SC)ccc1C(N1CC(O)(C(C)NC(c2nccnc2C)=O)C1)=O 41767,C1(C(N(C2CCCN(C(c3sc(C)nc3C)=O)C2)CC)=O)CC2(CCC2)CO1 41768,Cc1cccc(CN(C(=O)C(c2cccs2)NC(=O)C(C)n2ccnn2)C)c1 41769,c1(C(=O)NC2CC(N(C)C(C3CCC4(CCC4)C3)=O)C2)ccncc1N=[N+]=[N-] 41770,c1(C(N2CCN(C(C(C(=O)OC)C)=O)CC2)=O)nc2ccc(F)cn2n1 41771,C1(C(N2CC(N(C(=O)CCSc3nnnn3C)C)C2)=O)CCn2nccc2C1 41772,C1(C(=O)NC(CC2CCC2)CO)CCN1C(=O)C=C1CCC1 41773,C1(CNC(c2nc(COC)sc2)=O)CCCC(CNC(=O)C=CC=C(C)C)C1 41774,C(=O)(CCCC(=O)NCC1CCN(C(c2ccnn2C(F)F)=O)C1(C)C)OCC 41775,C1(NC(C2(CC#C)CCC2)=O)CCCC(NC(c2cc(C)n(C)c2)=O)C1 41776,Cc1nc2cc(C(=O)NCCCNC(=O)C(C)c3cccs3)ccc2n1C 41777,c1(C(C(=O)NCCCF)N(CC#N)CC)ccc(F)c(F)c1F 41778,C1(CC)CCC(C(=O)NC23CC(C(=O)NCC(F)(F)CO)(C2)C3)CC1 41779,C1(CCNC(C(C2CCOC2)OC)=O)CN(c2nc(C(C)C)ns2)CCS1(=O)=O 41780,c1(OCC=C)ccc([N+](=O)[O-])c(C(=O)NCC2CC2NC(=O)C(C)=CCC)c1 41781,Cc1nn(CC(=O)NCC2CC(C)N(C(=O)C=CSc3nc[nH]n3)C2)c(C)c1Cl 41782,C1(N(C(C(C(C)O)NC(c2cc(CC)on2)=O)=O)C)CCOC(C)(C)C1 41783,C1(C(N2CC3C(CNC(c4c(CC)scc4)=O)(C3)C2)=O)CC(C2CC2)=NO1 41784,C(C(=O)NC12CC(NC(c3csc(Cl)c3)=O)(C1)C2)(C(C)(C)C)NC(C)=O 41785,c1(C(=O)NCC2C(C)CCN2C(=O)C(F)=CCCF)cnn2c1OCC2 41786,CCC(CC)CC(=O)NCC1CN(C(=O)CCc2ccc(C#N)cc2)C1 41787,N1(C(C(CC)C)=O)CCCC(C(N2CCCC2Cc2ccccc2)=O)C1 41788,N1(CC(c2cc(F)cc(F)c2)C)Cc2ncn(C)c(=O)c2C1 41789,C=CCCCCCC(=O)N(C(C)C(=O)NC1CCCC(CC)C1)C 41790,C1(C(=O)NCCC(C)N(CCC)C)COCCN(C(=O)OC(C)(C)C)C1 41791,N1(C(C=C(C)C2CC2)=O)CC2C(N(C)C(c3ccc(-n4cnnn4)cn3)=O)C2C1 41792,CCCCCC(F)C(=O)N(C)CC.N1(C(C)=O)c2ncccc2NC1 41793,n1(CC)ncc(=NC(=O)C(CC2CC2)CC2CC2)[nH]1 41794,c1(NC(N)=O)cccc(C(=O)NC2CCCCC2CNC(C2CCCCO2)=O)c1 41795,CC1(C)Cc2occc2CN(C(=O)CC(N2CCOCC2)c2cccs2)C1 41796,c1(CNC(C2CN(C(C3(CC)CC3)=O)CCC2(F)F)=O)ccc(S(N)(=O)=O)cc1 41797,C1(C(=O)NC(C(C(C)C)NC(CN(C2CC2)CC)=O)C)CC2(C1)CC21CCC1 41798,c1(CCC(=O)NC(C2(O)CCN(C(CCOC(C)=O)=O)C2)C)c(F)cccc1F 41799,C1(OCCn2cc(COCC)nn2)CCCC(C(=O)OC(C)(C)C)CC1 41800,C(CC(O)CNC(=O)CNC(=O)CN(C)C)OC 41801,C(=O)(C(C)N(OC)C(=O)C=CC(C)NC(=O)C(C)NC(=O)C1CC1)OC 41802,N1(C(CCn2c(C)cc(C)n2)=O)CC(C)(C)CC1CNC(c1cc(Cl)sc1Cl)=O 41803,N1(C(C2(CC)CN(C(C(C=CC)O)=O)C2)=O)CCC(O)(COC)C1 41804,c1(C(=O)NCC(C)NC(CC)=O)cc(-c2ccccc2)n[nH]1 41805,C(=O)(CS(=O)(=O)CCC(F)(F)F)N(C(C)CCNC(C1CCCCS1(=O)=O)=O)C 41806,Cc1nc(C)c(C(N2CSCC2C(=O)NC(C2CCC2)C)=O)o1 41807,C1(NC(CNC(CC)=O)=O)(CNC(c2nn[nH]c2Cl)=O)CCOCC1 41808,Cc1ncncc1C(=O)NC1CCCC1CNC(=O)C(C1CC(F)(F)C1)O 41809,C1(CC(=O)NOCC2CCOCC2)CCCN(C(c2cn[nH]c2)=O)C1 41810,C#Cc1ccc(OC)c(C(=O)NCC2(C)CC2C)c1 41811,C1(=O)C(CCNC(c2ccoc2)=O)OC2CC(C2)N1C.CCS 41812,N1(C(C2(NC(C=Cc3ccc(C)o3)=O)CC(F)C2)=O)CC(C)OC2(CCC2)C1 41813,N1(C(C2C(CNC(C=C3CCC(C)CC3)=O)CCO2)=O)CC(C)C(O)C(C)C1 41814,CC1(CCNC(=O)Cn2cnnn2)CCN(C(c2ncncc2F)=O)CC1 41815,CC1CC(CO)CN(C(=O)C(C)NC(c2ncccc2Cl)=O)C1 41816,C(=O)(C(C)CC(N)=O)NCC(COC)NC(C(CCC)NC(C)=O)=O 41817,CCN=c1ccc(C(=O)NC2COCC2CNC(c2cccc(F)c2F)=O)c[nH]1 41818,c1(N2CCN(C(C(=O)NC(C)CC(C)(C)O)=O)CC2)ccc2cnccc2c1 41819,CC1CN(C)CC(C(N2CCOCC(C(=O)NC(C)C(O)C(F)F)C2)=O)O1 41820,c12coc(c1)CNC2=O.C(=O)(C(O)CSC)NCC1CN(C(=O)OC)C1 41821,Cc1nn(C)c2ccc(C(=O)NCC3CN(C(=O)Cc4ccco4)CC3O)cc12 41822,c1(C(N(CCCCNC(C(CC)O)=O)C)=O)c(C)sc(C)c1C#N 41823,c1(C(N(CCNC(C(c2cccnc2)OC)=O)C(C)C)=O)cnn2ccccc12 41824,c1(C(N(CCCCNC(c2ccc(C(N)=O)cc2)=O)C)=O)cccc2c1NCC2 41825,N1(C(c2ccc(CCC)cc2)=O)CC(C)(C)OC2(C1)CN(C(C1(O)CCC1)=O)C2 41826,Cc1cncc(CC(=O)NC(C2CCCN2C(C2COCCO2)=O)C)c1 41827,N1(C(C(CC)OC2CCCCC2)=O)CC2(NC(c3ncncc3C)=O)CC1C2 41828,CC(C)CC(CNC(C1Cc2nccn2C1)=O)C(=O)NCCC(C)C(F)F 41829,C(=O)(C(CNC(C1(C)CC=CC1)=O)CCC)NCCCSC 41830,CCC(C)C(C)CNC(C1CC=CC(NC(c2ccoc2)=O)C1)=O 41831,C(=O)(C#CC1CC1)NCC#CCNC(c1nc(CS(C)(=O)=O)sc1)=O 41832,C1(NC(CC2CCCC(C)(C)C2)=O)CC12CCN(C(=O)Cn1cnc(=N)[nH]1)CC2 41833,N1(C(C=C(C)C(C)C)=O)CCCC(C)C1CNC(c1cn(CC(F)(F)F)nn1)=O 41834,C1(NC(C23CC(C)C2C3)=O)CCC2CN(C(c3cccc(B(O)O)c3)=O)CC12 41835,C1(NC(C(COC)N(C)C)=O)CC(OC)CN(C(=O)CSC(F)(F)F)C1 41836,c1(OC)cccc2c(CC(=O)NCC(O)CCNC(=O)CO)c[nH]c12 41837,c1(CC(=O)NC2(CNC(C=CCCC)=O)CCCC2)cc(OC)cc(OC)c1 41838,C1(NC(c2c(CC)nccn2)=O)CN(C(c2cc(CO)ccn2)=O)CC1N=[N+]=[N-] 41839,N1(C(c2ccc(COC)s2)=O)CC2(CCC2NC(=O)C(C)(C)CSC)C1 41840,N1(C(c2nc(C#C)sc2)=O)CC(CNC(=O)COCCOCC)CC1(C)C 41841,c1(OC(C(=O)N(C(CCNC(CNC(=O)OC)=O)C)C)C)ccccc1 41842,c1(C(=O)NCCCC(C)NC(=O)C2=NNC(=O)C2)cc2cc(Cl)cnc2o1 41843,N1(C(c2c(C)[nH]nc2CO)=O)CCC2(CC1)CCN(CCC1CCCC1)C2 41844,C1(C(N(C2CCN(C(c3nn[nH]n3)=O)CC2)CC(C)C)=O)(CN)CC2C=CC1C2 41845,CC1OC2(CNC(C3CC3F)=O)CC1(NC(c1nccc(F)c1Cl)=O)C2 41846,N1(C(C2C(C3C(C)C3)C2)=O)CC2CN(CCOC3CCC3)CC2C1 41847,N1(C(C(CC)NC(N)=O)=O)CC(CNC(C2CC(F)(F)C2)=O)C2CCCCC12 41848,C(C(CCC)CCO)NC(C(c1c(C)cccc1Br)NC(CC(C=C)C)=O)=O 41849,CC1=NOC(CC(=O)NC2(C(=O)Nc3[nH]ccc3)CC(O)C2)C1.C(N)=O 41850,Cc1csc(C(N2CCCC2CCNC(c2ocnc2C(F)F)=O)=O)c1 41851,c1(C(N2CCN(S(C)(=O)=O)CC2)C(=O)NC(CC)(C)C)noc2c(Cl)cccc12 41852,C(CN=c1[nH]c(=NC2CCC=CCC2)[nH]c2cc[nH]c12)N(CC(F)(F)F)C 41853,C(=O)(C(C#N)(CC)CC)NCCC1(OC)CN(C(C2CC(C(C)C)=NO2)=O)C1 41854,C1(OC)CC(NC(C2CC(F)(F)C2)=O)CN(C(C2CCN(C3CC3)C2=O)=O)C1 41855,CC1CCCC(C)N(C(C2CC3CCC(C2)N3C(c2ccncc2Cl)=O)=O)C1 41856,C(=O)(C#CC1CCOC1)NC(C(=O)N1CCC(NC(CC)=O)C1)CCC1CC1 41857,C1(CC(=O)N(CC(F)Cl)C)CC(F)CN1C(=O)C=CC1CCCC1 41858,Cc1ccc2occ(CC(=O)N(C3CN(C(=O)C4=CC5CC=CCC45)C3)C)c2c1 41859,Cc1nc(C)c(CC(=O)NC2CCN(Cc3cn(-c4ccncc4)nn3)C2)s1 41860,C(=O)(C(C(C)(C)C)C1CCC1)NCC(C)NC(=O)C(C)S(C)(=O)=O 41861,N1(C(C(c2cnn(C)c2)OC)=O)CCCC(O)(CCNC(=O)CC(F)(F)Cl)C1 41862,O=C(N=c1[nH]oc2cccnc12)C1CCN(Cc2cnc(Cl)c(Cl)c2)CC1O 41863,Cc1c(Cl)ccnc1C(N1CCCCC1CNC(C1(N=[N+]=[N-])CC1)=O)=O 41864,N1(C(=O)OCC=C)CCCC(Oc2ccnc(O)c2)C1.C1(=O)NCCN1 41865,C1(N(CCCCC)CCC(=O)NC)CCN(C(=O)C(F)C(C)C)CC1 41866,Cc1cccnc1C(=O)NC1CC(F)(CNC(=O)C=Cc2cscn2)C1 41867,C1(NC(Cc2cccc(C(N)=O)c2)=O)CS(=O)(=O)C2CN(C(=O)CC3CC3)CC12 41868,c1(C(=O)NCC(C)CNC(C2CCC2(F)F)=O)cc2c([N+](=O)[O-])cccc2[nH]1 41869,CCC(C)C(O)C(=O)NNC(=O)c1ccc(C(=O)OC(C)(C)C)nc1 41870,C(=O)(CCCCC(=O)c1ccccc1)NC(C1OCCN(C(C(C)OC)=O)C1)C 41871,C#CC1CCCCN1C(C1CN(C(=O)CCC(=O)NCCC)CC1CCC)=O 41872,c1(CNC2CC(C(N3CCCC(CO)C3)=O)C2)cc(Br)ccc1Cl 41873,CCCCCCCC(=O)NC(CCCOC)C(=O)NCc1cn(C(C)C)nn1 41874,CCCCC(C)CCC(=O)N1C(C(=O)NCCOC2CC2)CCC1C(C)C 41875,c1(C(C(=O)NCCCOCCNC(C2(CO)CCC2)=O)OC)cnn(C)c1 41876,N1(C(C=CC=CCC)=O)CC2CC(C(N3CCSCC3C3CC3)=O)CC2C1 41877,C1(C(=O)NCC(C)N(C)C(c2ccc(F)o2)=O)CCC2(CC1)NC(=O)N(C)C2=O 41878,c1(SCC)ccc(CC(=O)NC(CCNC(c2ccsc2SC)=O)C(C)C)cc1 41879,c1(OC)ccc(F)c(C(=O)NC2CCCN(C(=O)Cc3cnnn3C)C2C)c1F 41880,C(c1ccc(Cl)s1)=[SH]CC(N1CCC(C(N2CCC(CC3CC3)CC2)=O)CC1)=O 41881,N1(C(c2ccnn2CCOC)C(=O)NC)CC2CC(O)C(O)CC2C1 41882,N1(C(CC(C)n2ccnc2)=O)CCC(C)(NC(C2CCC=CO2)=O)CC1 41883,CC(F)(F)C(C)(C)C(=O)N1CC(NC(c2ccc(N)cn2)=O)C(C2CC2)C1 41884,c1(C2(C)CC2)ccc(C(N2CC(O)(CNC(C3CC(C)(C)CO3)=O)C2)=O)cc1 41885,N1(C(C(C)Cc2ccc(O)cc2)=O)CCC2(CC1)CN(C(C1(C)CCCO1)=O)C2 41886,C(=O)(C(C)C(C)C)NCCCNC(COC(CC)(C)C)=O 41887,N1(C2CCN(C(C(C)C#N)=O)CC2)CCN(S(N)(=O)=O)CC1 41888,N1(C(CC2(N(C(Cn3nnc(C)n3)=O)C)CC2)=O)CCOC(C)C1 41889,C1(C(N2CC(N3CCCC3)C2)=O)CCCCCCN1C(C1CCCOC1)=O 41890,c1(C(=O)NCCCCCCNC(C2CCS2(=O)=O)=O)ncnc(O)c1Cl 41891,C#CCC(CC(F)F)NC(C1CC12CCN(C(C1(C)CC=CCC1)=O)C2)=O 41892,C1(C(=O)OC)CCC(CNC(CC2CC2)C(=O)N2CCC(Cc3ccoc3)C2)O1 41893,N1(C(CSCC=C)=O)CC(CNC(=O)COC(F)F)OC2(CCC2)C1 41894,c1(C(=O)NC(c2nc(C)[nH]n2)C(C)C)nsc2cc(Br)ccc12 41895,C12(C(=O)NC(C)C#N)CCC1CN(C(C1CCNC(=O)C1)=O)C2 41896,Cc1cccc(C(C)C(=O)N2CC(CN(C(=O)C=CCF)C)C2)c1.CC(F)(F)F 41897,c1(C(=O)N)ccnnc1O.c1(C(C)N(C(CC(C)F)=O)CCO)ccc(C(C)(C)C)cc1 41898,N1(C(C=CCN(C)CC)=O)CC2CC(NC(=O)CC(C)(C)C3CC3)C1C2 41899,c1(C(N2CCCN(CCNC(C(CC)F)=O)CC2)=O)cccc2c1CCCN2 41900,CC1CN(C(C2CNC(=O)N2)=O)CC1(C)C(=O)NC1CCNC(=O)CC1 41901,Cc1scc(C(=O)NCC(C)N(C)C(c2csc(CC(F)F)n2)=O)c1C 41902,C1(C(=O)NCCN(C(=O)Cc2csnc2C)CCC)CC12CCC(C)(C)CC2 41903,CC1(NC(C2CC3(CCC3)CO2)=O)CCN(C(=O)COc2ccon2)CC1 41904,N1(C(C(COCC)C)=O)CCC(CNC(=O)Cc2n[nH]c(=N)s2)(COC)CC1 41905,C(=O)(CCCCC(N)=O)NC1CCC(C)(CNC(C2(CF)CC(F)(F)C2)=O)CC1 41906,CCCC(CC(C)C)C(=O)N(CCNC(c1cc(N(C)C)ccn1)=O)C1CC1 41907,N1(C(c2n(CCC)ncc2)=O)CCC2(C=C(C(=O)N3CCC(OC)C3)C2)C1 41908,C#CC1(C(=O)NCC2(C)CCCN(C(C3(O)CCC3)=O)C2)CCOCC1 41909,N1(C(c2cc(F)c(F)c(F)c2)C(=O)NCC2CC2)CC2C3C=CC(C3)C2C1 41910,C1(C(=O)OCC)(C(=O)NCC)CC(O)C1.C1(N(CC(=O)OCC)C)(CO)CCOC1 41911,N1(C(C(CC)N(C)C)=O)CC2CN(C(=O)C(C)CSC)CC2C1 41912,Cc1cc(C(N2CCCC(NC(=O)C(C)(C)OC(C)C)CC2)=O)c(F)cc1F 41913,CCC(C)CC(C)C(=O)NCC1(CNC(=O)CCCCC(C)C)CCCC1 41914,N1(C(C(C)=CC2CC2)=O)CCOC(C)(CNC(c2cc3sccc3s2)=O)C1 41915,C(CCCC(C)(C)C(=O)NNC(=O)C1CCC(O)C1)NC(C(CC#C)O)=O 41916,Cc1cnnc(O)c1C(=O)NCc1nc(CNC(c2c[nH]nc2Cl)=O)cs1 41917,Nc1cc(C(=O)NCC2CCN(C(C34CCCN3CCC4)=O)CC2)cc(O)c1Cl 41918,C1(NC(c2c(Cl)cn(CCC)n2)=O)CCN(CC=C(Cl)Cl)CC1C 41919,c1(C(C)(C)C(=O)NC2CCCC2CNC(=O)Cc2cnco2)ccc(O)cc1 41920,Cc1cc(-n2nc(C3CSC3)nc2CC2CCOC2)cc(Br)c1 41921,c1(C(C(=O)NC(CNC(c2c(CC)con2)=O)C)(C)C)ccc(F)cc1F 41922,c1(CN2C(C(N3C(C)CCC3CO)=O)CC3CC32)cc(F)c(Cl)c(F)c1 41923,CC(C)CC(O)C(=O)N(CCC(=O)NC1CC2CCC1(CO)C2)CCO 41924,C1(NC(COC2(C)CCC2)=O)CCCN(C(c2ccc([N+](=O)[O-])o2)=O)CC1 41925,C1(C(=O)NCC(C)CO)CCN(C(c2ncn(C)n2)=O)C(C)(C)C1 41926,N1(C(CCCOCCOC(C)=O)=O)CCC2CN(C(c3ccc(C)nn3)=O)CC2C1 41927,C(=O)(C(F)C(F)(F)F)NC(c1cn(C)nn1)C(=O)N(C(CC)C1CC1)C 41928,C12(COC)CCC(C(=O)NCC3C4CN(C(=O)C=C(C)Cl)CC34)(CC1)CO2 41929,c1(C(=O)OCC)c[nH]c(=NC2CN(C(C3CC(C(C)(C)C)=NO3)=O)CC2C)cn1 41930,c1(C(C(=O)N(CCN(C(=O)CC2CC=CCN2C)C)C)O)ccc(Br)cc1 41931,N1(C(CC(=O)N(C)C)=O)CC2CC(NC(=O)C(c3ccccc3)N(C)C)CC2C1 41932,C(C(C(=O)NCCNC(=O)CC1CSCN1C(C)=O)OC)OC 41933,N1(C(C2C(C)C2C)=O)CC2CCCC(NC(c3ccc(C(N)=O)c(Cl)c3)=O)C2C1 41934,CC(C)C#CC(=O)N(C1CCCCC1)CCNC(=O)C(n1ccc(Br)n1)C 41935,C1(C(=O)NC2CC(CC(=O)NC3CC(C(C)O)C3)C2)CCCC12CCC2 41936,C1(NC(c2c(C(=O)OCC)cn(C)n2)=O)CCC(O)CN(C(=O)C(C)SC)C1 41937,N1(C(c2cnc(SC)s2)=O)CCCC2CCN(C(=O)Cc3ccn(C)n3)CC12 41938,C1(C)(CNC(CN(C(=O)C(O)C2CCC2)CC)=O)CCCCO1 41939,N1(C(c2c(-n3cccc3)sc(C)c2C)=O)CCCN(C(=O)CCC(N)=O)C(C)C1 41940,C1(C(=O)NC(C(=O)NCC)C)CC(C)CCN1C(C1CC2(CCC2O)C1)=O 41941,N1(C(c2cn(C)nn2)=O)CC2C(C(=O)N(C3CCCC3)Cc3ccccc3)C2C1 41942,c1(C(N(CC(C)O)CCNC(CC2(OC)CCC2)=O)=O)cc2scnc2[nH]1 41943,C(=O)(C1CCc2cccnc21)NCC1(C)CCN(C(=O)COC2CCOCC2)C1 41944,CC(C)CC(F)C(=O)NC1COCC1CNC(c1coc(C(C)(C)C)n1)=O 41945,N1(C(CC(C)NC(=O)C(N)=O)=O)CC(Nc2ccccc2C(N)=O)CC2(CC2)C1 41946,CC(C)CCCC(=O)N1CCN(C(=O)C=CCO)CC1CO 41947,C1(CNC(C(C)(C)OCC)=O)CC(C)N(C(c2cccc(-n3cccc3)n2)=O)C1 41948,c1(OCC)ccc(OCCC2CCCN2C)c2ccccc12.C1C(=O)N1 41949,N1(C(C2N(C(C)C)CCCC2)=O)CC2(CCN(C(=O)CC3(CO)CCC3)CC2)C1 41950,C1(CC(=O)N(C(CNC(c2cc[nH]n2)=O)Cc2ccccc2)C)CCC=CCC1 41951,C1(CNC(c2cc(C)c(C)[nH]2)=O)CC2(CC2)CN1C(=O)C(C(C)C)NS(C)(=O)=O 41952,N1(C(c2cn(C)nc2)=O)CCC(C(=O)Nc2ncc(F)cc2F)C(O)C1 41953,C(C(=O)NC(C(=O)NCCNS(N)(=O)=O)C1(C)CC1)(C(C)C)OCC 41954,c1(C(N(C2CCN(C(=O)C=Cc3ncc[nH]3)C2)C)=O)ccc2cnnc(O)c2c1 41955,c1(C(=O)NCC2N(C(C(C(C)(C)O)F)=O)CCC2)cc2c(O)cccc2[nH]1 41956,C#CC(C)(C)C(=O)N1CC(=O)CC1C(N1CCC(CC)C1)=O 41957,c1(C(=O)NCCC(C)(C)NC(CSC)=O)ccc(S(=O)(=O)N2CCCCC2)o1 41958,n1(CC=C)cc(C(=O)N(C2CCCC2)CCNC(=O)CSCCC(F)(F)F)nn1 41959,c1(C(C)=O)cn2c(n1)CN(C(=O)CCCOc1ccc(NS(C)(=O)=O)cc1)CC2 41960,c1(CN(C(CCC=C(C)C)=O)C(=O)C(O)Cc2cnc[nH]2)cccc(C(C)C)c1 41961,C1(NC(C=COCC)=O)CCC2CCN(C(=O)CC(C)n3cccn3)C1C2 41962,N1(C(c2cnc(C)s2)=O)CC(NC(C2(C)COC2)=O)CC(O)C1 41963,c1(C(=O)NC(CNC(CCc2n(C)ccc2)=O)C2CC2)coc2ccccc12 41964,N1(C(Cc2nc(C)sc2C)=O)CC2CCCC(NC(=O)CC3(O)CCCC3)C2C1 41965,C12(C(N3CC=CC(NC(C4C(C(=O)OC)C4)=O)C3)=O)CC(C)(C1)OC2(C)C 41966,c1(C(=O)NC(c2cc(F)cc(Cl)c2)CNC(CC2C(CC)C2)=O)cc(C#N)cn1C 41967,N1(C(C(CC2CC2)OC)=O)CCC(N(C)C(c2cc(N)c(C(=O)OC)s2)=O)CC1 41968,c1(C(N2CC(F)CC(NC(=O)CC3CC=CC3)C2)=O)cc2cc(Cl)ccc2o1 41969,C(=O)(C(CC(C)C)NC(=O)OC)N(CCNC(c1sc(O)nc1O)=O)CC 41970,N1(C(c2cc(C)nc(C)c2)=O)CCOC2(C1)CN(C(=O)C(C)OC1CCOC1)C2 41971,N1(C(CC(CCC)C)=O)CCC2(C1)CN(C(C1CCCN1c1cnccn1)=O)C2 41972,C1(C(N(CC(C(C)C)C)C)=O)C(C)OCCN1C(c1c[nH]c(=O)cn1)=O 41973,C1(NC(C2C(C)CCO2)=O)(CNC(=O)CN(C2CCCCC2)C)CCCCC1 41974,c1(CC)nccnc1C(=O)NCC(N1CCN(C(=O)C(O)C(C)SC)CC1)=O 41975,C1(CC)CN(C(C2(CO)CCOCC2)=O)CCC1NC(c1ns[nH]c1=O)=O 41976,c1(C(=O)NC(c2ccccc2)CNC(C2(CF)COC2)=O)cccc2nc[nH]c12 41977,C(=O)(CC(C)CC(=O)N1CCCN(C(=O)Cc2ncc(Cl)s2)CC1C)OC 41978,c1(-c2ccc(OCCOCC)cc2)cncc(F)c1C(=O)NCCC#N 41979,c1(OC)c(C(=O)N(CC(C)CNC(c2nocc2C(C)C)=O)C)cc(Cl)cc1Cl 41980,N1(C(C2CC(NC(c3c(CC)ncs3)=O)C(O)C2)=O)CCS(=O)C(C)C1 41981,C1(NC(C2CC(N(C)C)C2)=O)CCCCN(C(=O)Cc2ccc(Cl)c(F)c2)C1 41982,C1(NC(Cc2c(C)ocn2)=O)CN(C(C2CC3CCCCCC23)=O)CCC1(C)C 41983,N1(C(CC2OCCN(C(c3c(C)ccnn3)=O)C2)=O)CC(O)CC(C)(C)C1 41984,C1(NC(=O)Nc2cc(C)c(-n3cccn3)cc2)C2Cc3ccc(Br)cc3C12 41985,c1(OC)ncc(Br)cc1CN1CCOCC1CC(=O)Nc1ccc(C)cc1OC 41986,c1(C(=O)NC(C2CCCN2C(=O)CNC(N)=O)(C)C)coc2c1C(=O)NCCC2 41987,N1(C(C(=CC2CCCC2)C)=O)CCC(NC(c2sccc2C2CC2)=O)C(CO)C1 41988,c1(-c2c(C(=O)Nc3cccc(C(N)=O)c3)csc2)ccc(Br)c(OC(F)(F)F)c1 41989,C1(CNC(c2nccc(C(=O)OCC)c2)=O)CCC(C)CN1C(=O)C(O)C1CC1 41990,N(C1CN(C(=O)Cn2cncn2)CCc2ccccc21)C(C1=CC(C)(C)C1)=O 41991,Cc1nc(=NCC2CCCCN2C(c2ccc(C3CC3)cc2)=O)[nH]cc1[N+](=O)[O-] 41992,CC(CC(=O)NCc1ccnc(C(N2CCCC2(C)CO)=O)c1)CC(C)(C)C 41993,C1(NC(CCCC)=O)COCCN(C(=O)CNC(=O)CCC(C)C)C1 41994,N1(C(C2N(C(CC)=O)CCCC2)=O)CC(NC(=O)CC(C)(C)O)C2CCCCC12 41995,c1(C(=O)NCC2(C)CCCN(C(CCC(C)(C)F)=O)C2)ccc2nc(O)oc2c1 41996,C(C)(CNC(=O)COc1ccc(CCOC)cc1)(C(C)C)NC(C=C(CC)C)=O 41997,NS(=O)(=O)c1ccc(C(N2CC(CC(N3CCN(CCCO)CC3)=O)C2)=O)o1 41998,CC(C)CC(C)CN=c1[nH]c(N2CCC(C3CCN(C)C3)CC2)nc2c1CSC2 41999,C(=O)(CCC(C)(C)[N+](=O)[O-])N(CCC(C)C(F)F)C.C1(=O)C(C)(C)CN1CC 42000,CC1COC(CC(F)(F)F)N1C(=O)Nc1ccccc1-c1cccnc1 42001,N1(C(c2cn(C3C=CCCC3)nn2)=O)CCN(CC(F)(F)F)CC1.CC(C)(C)O 42002,N1(C(c2c(OC)n[nH]c2)=O)CCN(C)C(C(=O)NC2CCNC(=O)C2)C1 42003,C1(NC(C2C(C)(C)C2)=O)CCCN(C(c2cc(Cl)nnc2Cl)=O)CC1 42004,Cc1ccc2c(c1)CC(C(=O)NC(CNC(=O)CCc1cnoc1)C1CCC1)O2 42005,Cc1c(C(=O)NCC(C)(C)CNC(=O)C(C)NC=O)ccc(Br)c1F 42006,C1(N(C(=O)CSC(F)F)C)CCCCN(C(=O)C(C)(C)C2CCCC2)C1 42007,N1(C(CCNC(C2C(C)C2)=O)=O)C2CCC1CC(CNC(=O)CC1CC13CC3)C2 42008,N1(C(C(C(C)C)NC=O)=O)CC2(CCN(C(C3CC3(C)Br)=O)CC2)C1 42009,c1(C(=O)NC)cccc(C(=O)NCc2nc(CNC(C3COC(C)C3)=O)cs2)c1 42010,C1(C(N2CC(CCNC(c3c(C)nc(CC)s3)=O)OCC2)=O)CS(=O)(=O)CCO1 42011,N1(C(CCC(C)(C)C)=O)CC2CCN(C(=O)Cc3cccc4c3CCC4)CC2C1 42012,c1(C(=O)NCCC2CN(C(C(CC)OC)=O)CC2C)cnc2c(=O)[nH]ccc2c1 42013,C(CC)(C(=O)N1CC(N(C(=O)CCc2scnc2C)C)C1)=CC 42014,Cc1ccc(CNC(C2CC(C)(C)CN2C(c2cnn[nH]2)=O)=O)c(O)c1 42015,c1(C(=O)NC2CCC(CNC(C(C)O)=O)C2)ccc(OC(F)(F)F)cc1 42016,c1(CN(c2cc3ccccc3[nH]2)C)ccc2nccn2c1 42017,N1(C(CC(=O)NCC#C)=O)CCN(C(=O)CC2(CO)CC2)C(CCC)C1 42018,N1(CC)OCC(NC(=O)CC2CCN2C(c2cocc2C(N)=O)=O)C1=O 42019,N1(C(COCC(=O)NC)=O)CC(C)(C)OCC1CNC(C1CCCCCCC1)=O 42020,N1(C(C(C)CN(C)C)=O)CCN(C(C2(n3cncn3)CC2)=O)CC1CCN(C)C 42021,C1(C(=O)NCC2CC2CNC(c2coc(C)n2)=O)(OC)CCCOC1 42022,Cc1cn2c(n1)CCC(C(N1CC3(CCN(C(C4CC=CCC4)=O)C3)C1)=O)C2 42023,O=C(CS(=O)(=O)CCO)NCC1CCCC1NC(C1CNC(=O)O1)=O 42024,N1(C(C2C(NC(c3ccnc(SC)n3)=O)C2)=O)CC(F)(F)C(F)(F)C1 42025,c1(OC)ncc(C(=O)NC2CC(NC(=O)CC3CCOC(C(C)C)C3)C2)c(C)n1 42026,CC(C)CC(C)CC(=O)N1CCC=C(CNC(c2cn(C(C)C)cn2)=O)C1 42027,N1(C(CCC(C)N(C)C(c2ccc(OCF)cc2)=O)=O)CC2(C1)CC(C)(C)C2 42028,N1(C(CC2CCCC(C)C2)=O)CC2(CC(NC(=O)CC=CC(C)(C)C)C2)C1 42029,c1(OC)cc(N2CCC3CCC(C2)N3C(C2CCCO2)=O)ccc1[N+](=O)[O-] 42030,C(=O)(C1=CC2CC(C1)CC2O)NC(C)CNC(=O)CCn1cccn1 42031,N1(C(c2cnc(C(C)(C)C)nc2)C(=O)NCC)CCn2c(cnc2C(F)F)C1 42032,c1(NC(C2N(C(C3=C(C)OCC3)=O)CC(F)C2)=O)ncc(C)cc1C#N 42033,c1(CCC(=O)NCC2C(NC(c3nnc(C)s3)=O)COC2)ccccc1Cl 42034,C=CC(C)(CC)C(=O)NCCC1(C)CCN(C(c2ccsc2CC(=O)OC)=O)C1 42035,N1(C(C(CC)Oc2ccccc2)=O)CCC(NC(=O)C(C)(C)n2cccn2)CC1 42036,C1(C#N)(C(N2CC(CNC(C3(C(=O)OC)CC3)=O)C2)=O)CC1C(F)(F)F 42037,C(=O)(C1=C(C)CCOC1)NC(C(=O)NCC(C)OCC#C)C1CC1 42038,c1(C(=O)NCC(C)(C)NC(=O)CCc2ccsc2)cc(F)c2ccccc2c1 42039,CC1(C)CC(N=c2cc(C(F)(F)F)nc(Cl)[nH]2)CN(C(=O)CCC2CC2(F)F)C1 42040,c1(N2CCC(CNC(C3C(CC)OCC3)=O)C2)nc(Cl)c(C#N)s1 42041,N1(C(COC(c2nccn2C)C)=O)CCC(C(C)NC(c2ccns2)=O)CC1 42042,C1(CNC(C2CCN(CC)C2)=O)CC2CCC1N2C(=O)CCCCOC 42043,c1(C(CF)NC(=O)C(=O)Nc2ccccc2)ccc(Cl)cc1.C1(N)CC1CN 42044,CC(C)(CCCNC(=O)C(CO)C(F)(F)F)C(=O)NCC12CCC(CC1)OC2 42045,c1(C(N2C(C)(CC(=O)NC3(C#C)CC3)CC2)=O)cc(C#N)[nH]c1C 42046,c1(N2CCCC(NC(N)=O)C2)nc2c(c(=NCc3ccc(Br)s3)[nH]1)COC2 42047,C1(O)(CNC(C#CCNC(C2C(C(C)(C)C)C2)=O)=O)CCCOC1 42048,c1(CN(C(=O)C(=O)NCC2CC2)CCOC)c(C)nn(C)c1C 42049,N1(C(C(CC)N(C)C)=O)CCCC2CN(C(=O)COC3CCOC3)CCC12 42050,c1(C(C)(C)C)cccc(OCC(N2CC(CNC(=O)COc3cnsc3)C2)=O)c1 42051,c1(NC(C2CCC3(CCCN3)CC2)=O)ccnc2c(Br)cc(F)cc12 42052,c1(C(=O)OCC2C(C(=O)OCCC)C2)ccc(S(C)(=O)=O)s1 42053,CC1(C)CC(NC(=O)C=CI)CN1C(C1CC12CC2)=O 42054,N1(C(C(c2ccccc2)=O)=O)CC2CC(NC(C3(C4CCCO4)CC3)=O)CC1C2 42055,C(=O)(C(C)(C)C(=O)N(C)CC1CCN(C(c2ccccn2)=O)C1)NC 42056,c1(C(C)C)nnnn1CC(=O)NCC(=O)NCC1CCN1C(C1(C)CC1(C)C)=O 42057,C#CCC(CC#C)C(=O)N(C1CN(C(c2ccc(S(C)(=O)=O)o2)=O)CC1(C)C)C 42058,C1(NC(c2c(F)cncc2Br)=O)CC2(C1)CN(C(=O)C(O)CC1CC1)C2 42059,n1(CC(=O)NCC(C)N(C(C=C(CC)CC)=O)C)cccc([N+](=O)[O-])c1=O 42060,CC1(C)CN(C(C2CCCCO2)=O)C1C1CCN(C(c2ccon2)=O)CC1 42061,N1(C(C2CCCN(C(N)=O)C2)=O)C2CCC1CC(CNC(C1CC=CCC1)=O)C2 42062,c1(OC)ncc(Cl)cc1C(N1CC(CNC(C2CCC(C)(O)CC2)=O)C(C)C1)=O 42063,O=C(O)CCCCCCCCCNC(=O)CCCSC(F)(F)F 42064,c1(NC(C(c2n(CCC)ncn2)N(CCC#N)C(C)C)=O)cc(OC)ccn1 42065,CC1CN(C(c2ccnc(O)c2F)=O)CCC1N(C(=O)C=C(Cl)Cl)C 42066,c1(C(=O)NCC(CN(C)C(C2(F)CC2c2ccccc2)=O)O)nnc(C(C)(C)C)s1 42067,c1(CC(N2CCOCC(NC(C(C(C)C)O)=O)C2)=O)ccc(C#N)cc1F 42068,c1(C(=O)NC(C(C)NC(=O)CC2CCCOCC2)CO)cnc2sccn12 42069,C1(NC(CC2(C)CCN(C(COCCCC(C)C)=O)C2)=O)CCC=CCCC1 42070,CCC(C)(CNC(=O)CCc1cccs1)NC(C1CC=CCC1)=O 42071,c1(-c2nc(C(C(=C)C)O)n(C(C3CC3)OC)n2)ccc(N(C)C)c(F)c1 42072,c1(C(=O)NCC(CC)NC(c2ccc(N)cc2Cl)=O)cc(P(C)(C)=O)ccn1 42073,Nc1ccc(C(=O)NC2(C3CN(C(C4CCN4C4CCCC4)=O)C3)CC2)cc1F 42074,Cc1n[nH]cc1CC(=O)NC1CC(C)(CNC(=O)C(C)OCOC)C1 42075,CC(C)(CN=c1nc(N2CCCC(C(C)(C)C)C2)c2c([nH]1)CCC2)C(N)=O 42076,C1(C(=O)NC2(C3CN(C(C4C(CC(C)(C)C)C4)=O)C3)CC2)CS(=O)(=O)CC12CC2 42077,C1(OC)CCn2cc(C(=O)NC3CCCC(CNC(c4cscn4)=O)C3)nc2C1 42078,C1(C(N2CCCC(N(C(=O)COCC3(F)CC3)C)C2)=O)CCOCC12CCC2 42079,C(=O)(CC(C(F)F)n1ccnc1)NC(C(=O)OCC)Cc1ccccc1Br 42080,CCCS(=O)(=O)CC(=O)NCC1CN(C(c2sc(C)c(C)c2C)=O)CC1O 42081,Cc1cccc(C)c1C(=O)NCC1C(CNC(=O)C(C)NCC(F)(F)F)C1(F)F 42082,C1(CNC(=O)CC2CC23CC3)CN(C(=O)Cc2ccc(O)c(Cl)c2)CCCO1 42083,N1(C(C(C(C)C)O)=O)CC(C)OC2(CCN(C(c3ccc(F)cc3O)=O)C2)C1 42084,c1(C(N2CCC(NC(=O)C(F)(F)C(F)(F)F)C2)=O)ccc2c(c1)CNC2=O 42085,c1(CC(=O)NCCCNC(c2scc(C(=O)OCC)c2)=O)cnn2ccccc12 42086,CC(C(C(=O)NCSc1ccccc1)N1CC(C)C(O)C1)=Cc1ccsc1 42087,N1(C(Cc2ccc(C)s2)=O)CCC(NC(c2cnoc2-c2cccs2)=O)C(F)C1 42088,c1(C(=O)NC(C)(C)CCNC(c2sccc2CO)=O)ccc2c(c1)CCN2 42089,C12(C(=O)NC(CC)CCOC)C(NC(c3cccc(C)c3F)=O)C3CC1C2C3 42090,C1(CNC(c2conc2CNC(=O)CC2CSC2)=O)CCCC12CC2 42091,c1(OC)nccc(C(N2CC(C(=O)NC3CCC(NC(N)=O)C3)C2)=O)n1 42092,CC1C(C(=O)Nc2cccs2)C(C)CCN1C(=O)COC(=O)C#CC1CCCC1 42093,N1(CC(=O)NCC(C2CCCCC2)NC(c2ccc(OC)o2)=O)CCC(F)CC1 42094,C1(O)(CCNC(c2c(C)cns2)=O)CCN(C(C2CCCC(O)C2)=O)C1 42095,C1(C2CCN(C(C3C(C(C)C)(CC)C3)=O)C2)CCCCN1CC1CCCC1(C)C 42096,C1(C(N2CCC(O)(CN(C(C(C)=CC)=O)C)C2)=O)Cc2cncn2C(=O)N1 42097,C(=O)(C#CC1(CC)COC1)NCC(CC)NC(=O)C=Cc1cccc(Cl)c1Cl 42098,C(=O)(C(CCC)NC(C)=O)NCC1(C(=O)NC(CC#C)CC)CC=CC1 42099,C1(NC(C2C(OC)CC2)=O)CCN(C(c2cnc(S)n2C2CC2)=O)CCC1(F)F 42100,c1(C(=O)NC(CC)CNC(=O)C=Cc2ncc[nH]2)cnc(O)n1CC 42101,C1(C)(C(=O)NC2CC3(CN(C(c4c(C)cccc4C)=O)C3)C2)CC(C(C)C)=NO1 42102,CC1(C)CCC(C)(C)c2cc(C(N3CC4CCS(=O)(=O)CC4C3)=O)c(Br)cc21 42103,N1(C(=O)OC(C)(C)C)CCC(c2ccc(C(=O)Nc3cnn(CCl)c3)cc2)CC1 42104,C1(C(N(C)CC2CCN(C(=O)CC#N)C2)=O)C2CCC1(c1cncs1)C2 42105,C1(n2cc(C3N(C)CCC3)nn2)CCCC(NC(=O)CC2CC=CCC2)C1 42106,CCC(CC(=O)NCCc1cnc(C)cn1)N(C(=O)CCCCSC)C 42107,C(C)(C(C)N=c1cc[nH]cc1S(=O)(=O)N(C1CC2(CC2)C1)C)n1ncc(C)c1 42108,c1(CN(c2c[nH]c(=NC)s2)CC)ccc(F)c(Oc2ccccc2)c1 42109,C1(F)(CNC(c2nc(OCC)sn2)=O)CCCN(C(C2CNC(=O)C2)=O)C1 42110,c1(CNC(=O)Nc2c(C#N)cc(CC)s2)ccc2ccccc2n1 42111,C12(C(=O)NC3CC(CC(C)(C)C)C3)CC(NC(=O)CSCC(N)=O)(C1)C2 42112,C1(C(=O)NC2CCC(CNC(c3nc(C)n(C)n3)=O)C2)(OC)CCCCC1 42113,c1(OCCN(C)C)cncc(C(=O)N(C2CCN(C(c3ccco3)=O)C2)C)c1.CO 42114,N1(C(C=CCOC)=O)CC(NC(=O)COc2cc(C)on2)CC(C)C1 42115,c1(C(=O)NC2(CC=C)CCC2)c(CNC(=O)C(C#N)CC)cnn1C 42116,C12(CNC(=O)COc3ccon3)CC(CN1C(=O)C=Cc1nccs1)C2 42117,CC1(C)CCC(NC(C2CC23CCOC3)=O)C(CN=c2[nH]nc(CO)s2)C1 42118,C1(CNC(C(C)=CC2CC2)=O)C(C)CCCN1C(c1cccnc1)=O 42119,C=C(C)C1OCCC1CNC(=O)C(O)C1CN(C(C2(C)CC3C=CC2C3)=O)C1 42120,N1(C(CCOCCC)=O)CCC(C(C)NC(=O)C(c2cncn2C)=O)C1 42121,C1(C)(C(=O)NC2C(OC)CN(C(C=CCOC)=O)C2)Cc2ccccc2N1 42122,C1(NC(C2C(C=C)C2)=O)(COC)CCN(C(c2cccc(-n3nnnc3O)c2)=O)C1 42123,c1(CNC(CCC2CC(NC(C3C(C(=O)OC)C3)=O)C2)=O)nn(C)cc1C#C 42124,C(c1ccc(F)c(F)c1)=CC(N1C(CN(C(=O)C2=CCCSC2)C)CCCC1)=O 42125,Cn1cncc1CC(=O)NC1CCCC1C(N1CC(N2CCNC2=O)C1)=O 42126,C1(C(N(C)Cc2scc(C)c2)=O)C=CCCN1C(C1CCSCC1)=O 42127,c1(CNC(c2c(CNC(C(CC3CC3)OC)=O)noc2)=O)ccnc(F)c1F 42128,c1(CC)c(C(=O)NC2CCCCC2CNC(C2(C)CC2)=O)ccn1C 42129,N1(C(C(C)C2CC2)=O)CCC(F)(F)C(NC(c2cc(OC(F)F)ccc2F)=O)C1 42130,Cc1c(F)cc(C(N2CC3C(C(=O)Nc4cnn5ccccc45)C3C2)=O)cc1Br 42131,c1(C(=O)NCC(CNC(C2(C#N)CC2)=O)O)nn2c(c1Br)OCCC2 42132,CCC(C)(C(=O)Nc1cccc(NC(=O)CC2C=CCCC2)c1)OC 42133,C1(CCC2N(C(C(=O)N(C)C)=O)CCC2)CCCCN1C(=O)C=Cc1cocn1 42134,C(=O)(C(C)(C)CF)NCC(CCOC)NC(C1(N2CCCC2)CCC1)=O 42135,Cn1ncnc1C(c1nnnn1C)NCC1(C2CC2)CCCO1 42136,C(=O)(CC(C)C(F)(F)F)N1C2C(NC(CCOCCCOC)=O)C(CC2)C1 42137,Cc1ccoc1C(=O)N(CC(=O)NC1CCC(CO)C1)CC(C)C 42138,c1(CCC(=O)N(C2CC(NC(CC=CC)=O)C2)C)cnn(C)c1C 42139,CC1(C)CN(C(=O)Nc2cnn(C(F)(F)F)c2)CCS1(=O)=O 42140,c1(CCC(=O)OCC)nc2cc(-c3cc(CO)ccc3F)ccc2o1 42141,CC(C)C(C(C)NC(=O)C=CCF)NC(c1cc(C2(C)CC2)on1)=O 42142,C1(C(=O)NCCC(=O)N(CC)CC)CC2CCC1N2C(c1cc2n(n1)CCO2)=O 42143,O=C1CC(C(=O)NCC2(C3CC3)CCCO2)N(C(=O)C(C2CCCCC2)=O)C1 42144,c1(C(=O)NCC2(C(=O)NCC(N(C)C)C3CC3)CC=CC2)ccc(CF)cc1 42145,C1(NC(C2(SC)CCC2)=O)CC(n2cc(-c3ncccc3F)nn2)C(O)C1 42146,C1(C(=O)NCC2(C(C)C)CCCC2)CN(C(c2ccc[nH]2)=O)C2(CCC2)C1 42147,O=S(=O)(c1cccc(=NC2C=CCCC2)[nH]1)NC1(c2ccc(F)cc2)CCC1 42148,c1(CCC(=O)N(CC(C)O)CCNC(=O)CP(C)(C)=O)ccc(Cl)cc1F 42149,c1(CC(=O)NCC(C2CCOC2)NC(CCC)=O)coc2cc(Cl)ccc12 42150,C=CC(C)CC(=O)N(C1(C(=O)NCc2ccc(Cl)cn2)CCC1)C1CC1 42151,C12(CNC(c3cccc[n+]3[O-])=O)CCCC(CN1C(C1CCCCC1)=O)C2 42152,C(C(CC(C)C)C(=O)N1CC2(CC(C)CO2)C1)NC(C1C(OCC)CC1)=O 42153,N1(C(CSCC#C)=O)CC(C2CC2C(N2CC(N3CC(O)C3)C2)=O)C1 42154,c1(C(=O)NC2(C)CCN(C(C(CCC)N(C)C)=O)C2)c[nH]c2ncccc12 42155,c1(C(=O)NC(CNC(CC(C=C)c2ccccc2)=O)CO)cc([N+](=O)[O-])oc1C 42156,C1(N(C(C2CC2(Cl)C(F)F)=O)CC)CCN(C(c2snnc2C)=O)CC1 42157,c1(C(N(C)CC2CCN(C(CC3(COC)CC3)=O)C2)=O)cncc(OC)c1C 42158,C1(NC(C(C)NS(CCC)(=O)=O)=O)CC(NC(=O)CCNC(C)=O)CC1O 42159,C1(c2n(CC)nnn2)(NCCOc2ccc(F)cc2)CCCSC1.c1snnc1C 42160,c1(C(=O)NCC2N(C(CN(C)CC)=O)CCCC2(C)C)ccc2c(c1)CCCC2 42161,N1(C(Cc2cnn(CC)n2)=O)CCC(C(C)C)C1C(=O)NOC 42162,C(=O)(C(O)CC(C)(C)C)NC1C(CNC(C2CC(C)OC(C)C2)=O)CCCC1 42163,C1(CC(=O)NCCC2CC(NC(C#CC(C)(C)O)=O)C2)CC2(CCOCC2)CO1 42164,N1(C(c2c(NC)snc2C)=O)CC(NC(=O)Cn2ccnn2)C2(CC2)C1 42165,c1(C(=O)NCC2CN(C(c3c(OC)n[nH]c3)=O)C(C)C2)nccc2[nH]ccc12 42166,c1(C(N2CCCC(NC(c3c(CC)onc3C)=O)C2)=O)c(C)nn2cccnc12 42167,Cc1ccc(Cl)c(Oc2cccc(CNC3(CNCC(=O)OC(C)C)CC3)c2)c1 42168,c1(CC(=O)NC2(C(=O)NCC3(OC)CC3)CC2(C)C)cnn(C)c1C 42169,c1(C(=O)NCCN(C(=O)C(N(C)C)N(C)C)CC(C)O)cccc(S(C)(=O)=O)c1 42170,C1(CC(=O)NC2C(CNC(=O)CNC(=O)Cn3cncn3)C2)CN2CCN1CC2 42171,C1(CNC(C=CC=CCC)=O)CCCCCN1C(=O)CC(C)(C)CNC(C)=O 42172,C(=O)(CCCCCCC)NCC(CC=C)C(=O)NCCCCS(C)=O 42173,C=CC1(CC(=O)NCC(c2ccccc2)NC(=O)CC2(O)CC2)CCCCC1 42174,CCCCC(O)C(=O)NC1COCCN(C(C2CCCCN2C)=O)C1 42175,C1(NC(=O)CCCn2c(O)nnc2O)COCCN(C(c2ccsn2)=O)C1 42176,c1(CN2CC(NS(C)(=O)=O)(COC)C2)ccc2cccnc2n1 42177,N1(c2nc(OCC)c(Cl)cn2)CCC2(NC(c3ncccn3)=O)CCCCCC12 42178,Cc1ccc(C(=O)N(CCCCCC(=O)NCC2CCC(F)C2)C)nc1C 42179,N1(C(C=C(CC)C)=O)CCN(C(C2(C(C)(C)O)CC2)=O)CC12CC2 42180,O=C1NCc2ccc(NC(=O)CC3CCCC(C(F)(F)F)C3)cc21 42181,c1(C(=O)NCC2N(C(C3CC(N(C)C)C3)=O)C3CCC2C3)ccc2ncnn2c1 42182,N1(C(c2cn(CC)nc2)=O)CCC2CCCC12C(=O)NC(C)Cc1nncn1C 42183,C(=O)(C1=CCCCC1C)N1CC(N(C(CSc2cccc(OC)c2)=O)C)C(F)C1 42184,c1(C(N2C(CNC(Cc3cc(C)[nH]n3)=O)CC(F)C2)=O)c(F)c(F)cc(F)c1F 42185,C(C(CC=C)C(=O)NCc1ncsn1)NC(C(C)=CC=C)=O 42186,c1(CCN(C2CCNC2)CC(=O)NCc2nn[nH]n2)ccccc1 42187,C1(NC(CC2C(CNC(=O)COc3cccc(O)c3)C2)=O)CCC2(CC1)N=N2 42188,c1(CC(=O)NC2CCN(C(c3cocc3C(=O)O)=O)CC2)ccccc1Cl 42189,CC1CCCCC1C(=O)NC(C1CN(C(C2(C)CC(F)C2)=O)C1)C 42190,Cc1nc(C(=O)N(CCC(C(C)C)NC(c2cnc(O)c(Cl)c2)=O)C)cc(O)n1 42191,c1(CC)ncccc1C(=O)NC1CC(CNC(=O)COCC2CC2)C1(C)C 42192,N1(C(=O)NCc2cccc(C)n2)CCC(F)(F)C2(CC1)NC(=O)NC2=O 42193,c1(C(N(C2CCC(NC(=O)CCc3ccco3)C2)C)=O)ccnnc1O 42194,c1(C(N2CC(N(C)Cc3nnc(CC)o3)C2)=O)ccc2cc(C)ccc2n1 42195,c1(C(C)C)ccc2occ(-c3nc(CN4CCOCC4)nn3C3CCOC3)c2c1 42196,N1(C(c2c(C)csn2)=O)CC(NC(=O)C(C2CCOCC2)C)CCC(O)C1 42197,CC1(C(=O)NCc2cccc(NC(=O)Cc3ccccc3)c2)CC(C2CC2)=NO1 42198,Cc1c(CC(=O)NC2CC(NC(=O)CC(C)F)C2)c(=O)oc2cc(O)ccc12 42199,C1(N(C)C)CN(C(C2CC23CC(NC(=O)CCCC2CCCO2)C3)=O)CC12CC2 42200,N1(C(c2c(CC)nn[nH]2)=O)CC(CNC(=O)Cc2c[nH]nc2O)CCC1C 42201,N1(C(C2OCC(C)(C)C2)=O)CC2(CC2)CC1CNC(c1cc2n(n1)CCC2)=O 42202,C1(NC(C2(C)CCCS2)=O)CCN(C(c2cnc(C3OCCO3)s2)=O)CC(O)C1 42203,c1(C(N2C(CNC(C(C(C)(C)C)O)=O)C3CCC2C3)=O)sc2ncccc2c1N 42204,CC1(C)CNc2ccc(C(=O)NCC(F)CO)cc21 42205,C1(OC)CCCC(NCC(=O)Nc2cccc(I)c2)C1 42206,C1(NC(Cc2cc(C)on2)=O)CCOC(CNC(=O)Cc2ccc(Cl)cn2)C1 42207,CC(C)C(C(=O)NCC(C)CN(C)C(C1CN(C)C1)=O)C1CCC1 42208,C1(NC(Cc2c(C)nccc2)=O)CS(=O)(=O)CC1NC(C1(CF)CC1)=O 42209,C1(NC(c2c(CC)scc2)=O)CCN(C(=O)C(C)(C)C2CCOC2)CC1(C)C 42210,C(=O)(CC(C)(O)C(F)(F)F)NC1CCC(CNC(CCN(C)CCO)=O)C1 42211,N1(C(c2cc(C)nc(O)c2)=O)CC2CCC(C1CO)N2C(c1ccnc(O)c1)=O 42212,C(CC)(CCC(=O)NCC1(O)CCSC1)NC(CCC#C)=O 42213,C1(C(=O)NCCCCN(C(CCCCCC#C)=O)C)CCc2ccc(F)cc2O1 42214,C(N=c1[nH]c(=NCC(C)C#N)[nH]c2cc[nH]c12)c1c(OC)ccc(F)c1 42215,c1(OC)c(NC(=O)C=C2CCN(Cc3c(Cl)ccnc3Br)CC2)cccc1C#N 42216,C1(C)(C(=O)NCCC(C)(C)NC(=O)C(C2(O)CCCC2)F)CC(C(C)(C)C)=NO1 42217,C(c1ccccc1F)=CCC(=O)NC1CN(C(C2(CCCC)CCC2)=O)CC1O 42218,CCC(C)(C)C(=O)C(=O)N1CC(C(=O)NCC2(CO)CC2)C(F)(F)C1 42219,c1(C(=O)NC2C(NC(c3c(C)n[nH]c3)=O)CCC2)cnc2c(c1)NC(=O)CN2 42220,c1(C(N2CC(O)(CN(C(CC=CC)=O)C)C2)=O)ccc2c(c1)CCCS2(=O)=O 42221,C1(OC)CC(NC(=O)C2=CCC2)C12CCN(C(=O)CC1(O)CCCCC1)CC2 42222,N1(C(C2(C(=O)OC)C=CCC2)=O)CC(C2(NC(=O)C=Cc3ccoc3)CC2)C1 42223,CON1CCC(N(C(=O)C(c2cn(C)nn2)NC(c2ccc(Cl)cn2)=O)C)CC1 42224,C1(CNC(CSC)=O)(CNC(C2CNC(=O)O2)=O)CCOCC1 42225,C1(NC(c2cc(SC)oc2C)=O)CCN(C(=O)C(C)NC(=O)C(C)(C)C)CC1F 42226,Cc1c(C(=O)NCCC2CC(NC(=O)C(C)c3cccs3)C2)cnn1CC(F)F 42227,N1(C(N2C(c3n(CC)cnc3)CCCC2)=O)CCCc2ccc(F)cc21 42228,C1(C(NOC)=O)CC(C)N1C(c1cncn1C)=O 42229,N1(C(c2nc(CC)sc2)=O)CCC(C2CCCN(C(C3(O)CC3(C)C)=O)C2)CC1 42230,C(=O)(C(C)C(C)(C)C)NC(C)CNC(c1cn(C)nc1C(C)(F)F)=O 42231,N1(CC(=O)NC(CNC(c2cc(C(C)=O)on2)=O)C)CCCCC1=O 42232,Cc1cn2c(=O)c(C(=O)N(CC(O)CNC(C3CCCS3(=O)=O)=O)C)cnc2s1 42233,c1(C(N2CCN(c3nc(COC)nc(Cl)c3)CC2)=O)cc2cc(C)ccc2cn1 42234,c1(NC(C(C2CN(C(=O)CCC3(C#N)CCC3)C2)OC)=O)cnc2ncnn2c1 42235,C1(C(N(C2C(C)CCC2)C)=O)CC(NC(=O)CCn2cnc(=N)[nH]2)CCO1 42236,N1(Cc2ccc(N3CCCC(C(=O)O)C3)o2)CCCc2ccccc21 42237,Cc1cc(CNC(C2CC(NC(C3(N(C)C)CCC3)=O)CCO2)=O)ncn1 42238,C1(CC)(CC)CNC(=O)C1NC(c1cc(OC)c(Br)s1)=O 42239,c1(OC)ccc(C(C)NCC2CC(F)(F)C2(C)C)c(OC)c1 42240,C(c1cc(C)ccc1OC)=CC(=O)NC(CCOC)CNC(=O)C(F)=C1CCC1 42241,c1(C(=O)NC(c2cccc(Cl)c2)CNC(CN(C2CC2)CC)=O)nc(C)nn1C 42242,N1(C(c2cccc(CC)c2)=O)CCC(F)C(NC(C2CCCCC2CC)=O)C1 42243,CCCCCC(O)CC(=O)N1CC(O)(CN(C)C(C2(C#N)CCN(C)CC2)=O)C1 42244,c1(CC)ccc(NC(C2C3CS(=O)(=O)CC23)=O)c(C)c1 42245,CC(C)CCCCC(=O)NC1(CNC(=O)C(C)C2CC2)CCCC1 42246,Nc1c(Cl)cc(C(=O)NCC2(F)CC(NC(C3CC3[N+](=O)[O-])=O)C2)cc1[N+](=O)[O-] 42247,N1(C(c2ccc(CC)cc2)=O)CCN(C(=O)CCc2cccnc2)CC1C#N 42248,Cc1nc(C)c(F)c(=NCC(C(C)(C)C)NC(c2cccc3c2C(=O)NC3)=O)[nH]1 42249,c1(C(N(CC(C)NC(=O)Cn2cc(C(N)=O)nn2)C)=O)csc(C(F)F)n1 42250,C1(NC(C2(COC)CCCC2)=O)CC(NC(=O)C(C)(C)Cn2cccn2)C12CCC2 42251,n1(CC(N2CCC(C)(CNC(CS(CC)(=O)=O)=O)C2)=O)cc([N+](=O)[O-])c(C)n1 42252,CN1CCOC(C(N2CCOC(C3CN(C(c4cnn(C5CC5)c4)=O)C3)C2)=O)C1 42253,N1(C(CN(C)C(N)=O)=O)CC2CCC(NC(c3c(Cl)ccnc3F)=O)CC2C1 42254,c1(C(CNC(CNC(CC2(N(C3CCC3)C)CC2)=O)=O)O)cnn(C)c1 42255,C12(NC(CCOCCCOC)=O)CCCN(C(C3(C)COC3)=O)CC1C2 42256,C(CN=c1[nH]c(=NC(C)c2ccoc2)c2sccc2[nH]1)c1c(C)nc[nH]1 42257,n1(CC)cc(Cl)c(C(=O)Nc2cccc(NC(=O)CCC3CC3CC3CC3)c2)n1 42258,C1(O)(CC#C)CCN(C(=O)C(C(C)CC)N(C(=O)CCCC#N)C)CC1 42259,C(CCCCCCCO)=CC(=O)NCC(CNC(C1(CCCC)CC1)=O)(C)O 42260,CC1C(NC(=O)CC2CCCC2)CC2CCC1N2C(c1ccc(C2CC2)o1)=O 42261,c1(C(=O)NC(CCC)CNC(=O)C(C)(F)c2ccccc2)cc(C)c(C)o1 42262,c1(OC)cc(F)c(F)cc1S(=O)(=O)N1CC(C)(C)CC1C 42263,C(CC(C)C)(C(=O)NC1(CO)CN(C(c2cccc(OCCO)n2)=O)C1)OC 42264,N1(C(C2C3CN(C(CC(C=C)CCC)=O)C2C3)=O)CCc2cc(C)ccc21 42265,c1(C(N(C(=O)CC2CCC(NCC3CC3)CC2)CCO)=O)cccc(OC)n1 42266,C1(NC(c2c(C)nsc2C)=O)CC12CCN(C(c1cnn3ccn(C)c13)=O)CC2 42267,N1(C(C(C2CCCN(C(C(CC)(C)COC)=O)C2)C)=O)CC(C)N(C)C(C)C1 42268,C(C(C)(C(=O)N(CC(C)(C)CO)C)NC(c1cc(=N)[nH][nH]1)=O)SC 42269,C1(C(=O)NC(C)(CO)CCF)CCCC(NC(=O)C=Cc2ccco2)CC1 42270,N1(C(C(C)NC(CC)=O)=O)CC2CC(NC(c3coc(C(C)C)n3)=O)CC1C2 42271,c1(NCc2c(C(C)(F)F)n[nH]c2)cc2c(cc1Cl)NC(=O)C2 42272,N1(C(C2CC(C)(C#N)C2)=O)CC2CCCC2(CNC(c2ccsc2Cl)=O)C1 42273,CCC(O)C(F)(F)C(=O)N1CC(CCNC(=O)C(CC)c2ccccc2)(OC)C1 42274,c1(C(=O)NCC(C)N(C(=O)CCCn2cncn2)CC)c(C)cccc1C 42275,C1(O)(CNC(C(CC)(C)F)=O)CCCN(C(=O)CN2CCCCC2=O)CC1 42276,N1(C(CC2(C)CC2)=O)C2CCC1CC(CNC(=O)CCCC1CCCC(=O)N1)C2 42277,C(CNC(C1(Cl)CC1(F)F)=O)(CC(=O)NCCc1cnn(C)c1C)OC 42278,C1(C(=O)NCC2CC(C)(C)CO2)(CC)CCN(C(C2CCCC3CC23)=O)CC1 42279,CCCC(C)(C)CC(=O)N1CCC(N(C(=O)CCOCC2CCC2)C)C(C)C1 42280,CCCCC(CC)CC(=O)N(C1CC(NC(c2csnn2)=O)C1)C 42281,CC1C(C)N(C(=O)C=Cc2ccco2)CCN1C(=O)C=Cc1ccc(C2CC2C)o1 42282,N1(C(c2c(CC)non2)=O)CC(NC(=O)Cc2ccc(C)cc2)C(C)C1 42283,C12(CCCCC1)CC(=O)NC2.C1(O)(C(C)NC(C)=O)CCN(C(C)=O)C1 42284,Nc1ccc(C(=O)NC(CNC(=O)C(O)C2CC2)CC(F)(F)F)c(Br)c1 42285,c1(OC)ccc(Br)c(C(N2CCC(N(C)C(c3ccccc3)=O)C2)=O)n1 42286,CCC(CC)C(=O)NCC(N1CCOCC1CNC(C1CCCC1)=O)=O 42287,C12(CCNC(c3cncc(C)c3)=O)CCC1CN(C(C1CCCN1C(N)=O)=O)C2 42288,C12(C(N3CC(CC(=O)OC)C3)=O)CC1CCN2C(c1ccc(CO)o1)=O 42289,c1(C(=O)NC2CCN(C(CCN3CCC(C)CC3)=O)C2)ccc2cc[nH]c2c1 42290,C(c1sc(Cl)nc1Cl)=CC(=O)NC1(COC)CCN(C(C23CCCC2C3)=O)C1 42291,N1(C(C2C(C)OCC2)=O)CCC(NC(c2c[nH]cc(Br)c2=N)=O)C(C)(C)C1 42292,c1(C(c2n(CCCOC)nnn2)NCC2CC2)ccc2c(c1)COC2(C)C 42293,CC(C)C(CCNC(C1(c2ccccc2)CC1(F)F)=O)NC(c1cncc(O)c1)=O 42294,Cc1cc(C(=O)NCC2CCN2C(c2ccc(CC3CC3)cc2)=O)nc(O)n1 42295,C1(c2n(C(CC)C)nnn2)(NCc2ccns2)CCCN(Cc2ccccc2)C1 42296,c1(NC(=O)CC2CC(NCc3cc(Br)cnc3F)C2)cc2ccccc2cc1O 42297,c12ncccc1C2.c1(NC2(NC(=O)CNC(=O)C(F)(F)F)CC2)ccsc1SC 42298,C1(N(C(C=Cc2n(CC)ncc2)=O)C)CCCN(C(=O)CC2CC2C2CC2)CC1 42299,CC(CC(=O)N(C1CC(NC(c2sc(Br)cc2Cl)=O)C1)C)C(F)F 42300,C1(C(C(=O)N(CC(C)NC(=O)CSC(F)F)C)OC)CCOCC1 42301,C(C(=O)C(C)(C)CC)OC(C(=O)NC(c1ccc(OC)cc1)CC)=O 42302,N1(C(c2c(COC)con2)=O)CCC2CN(C(C3(C(=O)OC)CC3)=O)CC2CC1 42303,C(CN=c1[nH]c(=NCC2(S(C)=O)CC2)[nH]c2c1CSC2)c1c(C)noc1C 42304,c1(C(=O)NCC2CC(NC(c3cc(COC)sc3)=O)C2)cnc(O)c(Cl)c1 42305,c1(OC)cnnc(C(=O)N(C)CCOC2(C(=O)O)CC2)c1 42306,N1(C(c2cn(C)nc2Cl)=O)CCN(C(C2(F)CCS(=O)(=O)C2)=O)CC1C1CC1 42307,c1(C(C(=O)NCC2CCCO2)N(C2(C#C)CC2)C)cc(Br)c(Cl)cc1OC 42308,Cc1ccnc(C)c1C(=O)OCCCNCC1CC1c1cnn(C2CC2)c1 42309,c1(C(=O)NC2C=CCN(C(C(C)OCCC=C)=O)C2)nc2c(s1)COCC2 42310,c1(C(C(=O)NCCCN(C(C)=O)C)NC(=O)COC(C)(C)C)cnc(O)nc1O 42311,C1(=O)NNC(=O)CO1.CC1CCC(C(=O)OC(C)(C)C)N1C(=O)C1=CCCC1 42312,N1(C(CCCn2cc(CCN(C)C)nn2)=O)CCCC(n2ccnn2)CC1 42313,c1(CNC(C2CC(CCC)C2)=O)cn(C2CCN(C(c3cnc(Cl)s3)=O)C2)nn1 42314,C(=O)(C(C)S(C)(=O)=O)N1C(C2CCCN(C(c3c(C)noc3C)=O)C2)CCCC1 42315,C1(C(N2CC(NC(C3C(C)(C)C3)=O)C(F)C2)=O)CC2(CCCO2)C1 42316,c1(C(=O)NCCC2(C)CCN(C(COC(C)=O)=O)C2)n[nH]c2ccccc12 42317,c1(NC(C)=O)cnc(O)c(C(=O)NCC2CCC2NC(C2(C)CC3CC3C2)=O)c1 42318,C1(NC(c2cc(CC)on2)=O)CC2(C1)CC2NC(=O)C(O)C(C)C 42319,CCC(C)C(C(=O)N(CCN1CCCC1)CC1CCCO1)NC(=O)NC 42320,Cn1cc(OCC(N2CC(C)(NC(=O)CCc3cscn3)C2)=O)cn1 42321,CS(=O)(=O)C1CN(C(=O)C(CC2CCC2)NC(=O)CC2CCCSC2)C1 42322,c1(CC)ccc(C(N2CCC2C(=O)NCC2(C#N)CC2)=O)cc1 42323,c1(OC)cnc(C(N2CC3C(CNC(=O)C=Cc4ccc(Cl)s4)C3C2)=O)c(F)c1 42324,c1(C(N2CCC(C(=O)NC(CCC)CO)C2)=O)cc2cnccc2nc1C 42325,c1(C(N2C(CNC(c3c(OC)ccs3)=O)CC2)=O)cc(C(F)(F)F)cc(O)c1 42326,C(C1CN(C(=O)CN2CC3CC3C2)CC1C(=O)NC1C2CCCCCC12)=CC 42327,c1(C(=O)NCC2CC(COC)CN2C(=O)Cc2cncnc2)cccn(C)c1=O 42328,CCCCCCCCCCS(=O)(=O)N1CCCC(CNc2ncc(CC)s2)CC1 42329,N1(C(CCC(=C)Cl)=O)CC(NC(c2n[nH]c3c2CC2CC32)=O)CC12CCCCC2 42330,C1(=CC(=O)NCC2C(NC(C3CC3CC(=O)OC)=O)C2)CCOCC1 42331,N1(C(c2cc(COC)[nH]n2)=O)CCCC1(C)CNC(=O)C#CC1CC1 42332,C1(C2CCCCC2)(C(=O)NC(CC(C)NC(c2cc(OC)no2)=O)C)CC1 42333,N1(CC(C)(C)N(CC(C)C)C(=O)OC(C)(C)C)CCC(C(C2CCCO2)C)CC1 42334,C1(CNC(C2(CC)CC2(F)F)=O)CCN(C(C2(C3CC3)CC2)=O)CC1C1CC1 42335,c1(C(c2nnnn2CCCF)NCC(C)(C)SC)cnn(C)c1C 42336,C1(OCC(=O)NC(C2CCCN2C(=O)C=Cc2c[nH]cn2)C)CC(F)(F)C1 42337,N1(C(c2cc(C)c(Cl)cc2)=O)CC2CCC(C1)N(C(=O)CCC(F)(F)C(F)F)C2 42338,c1(CC(=O)NCC(CNC(=O)C=CC2CCCC2)OC)ccccc1SC 42339,Cc1c(-c2cn(CCCC(=O)N(CC(N)=O)C)nn2)c(=O)oc2ccc(O)cc12 42340,C(=O)(CCCCCCN=[N+]=[N-])NC1C(C)CN(C(=O)CN2CC(C)(C)C2)CC1 42341,N1(C(C(CSC)O)=O)CCC2(CCCCC2NC(c2ncc(F)cc2F)=O)CC1 42342,c1(CCNC(C(=O)N(C(c2c(C)cccc2)C)C)=O)ccc2c(c1)CC(C)O2 42343,c1(N2CC(Oc3cccc(NC(C4CC(=O)NCC4)=O)c3)C2)ncnc2[nH]cnc12 42344,N(C(=NCCN1CCOCC1)NCC1CCC(F)C1)CC1(CS(C)(=O)=O)CCC1 42345,C#CC1(NC(=O)C(O)CCNC(c2cccc(=O)o2)=O)CCOC1 42346,C1(CCOC)CCCN(C(=O)OC(C)(C)C)C1.c12csc(n1)NC2 42347,C1(C)(C(=O)NCC(CN(C(=O)COC2(C)CCC2)C)(C)C)CCC(=O)NC1 42348,c1(C(=O)NCC2(OCC)CCN(C(CCC)=O)CC2)coc2cc(F)ccc12 42349,C(=O)(C1=CC2CC=CCC12)N1CC(NC(c2n(C)ncc2C2CC2)=O)C1 42350,CCC(O)C(=O)N1CCC(N(C)C(c2cc(-c3cccnc3)no2)=O)C1 42351,Cc1ccc(F)cc1C(N1CC2(CNC(c3cc(Cl)c(Cl)n3C)=O)CCC1C2)=O 42352,C1(NC(C2C(NC(C(CC)(C)C)=O)COCC2)=O)CCCOC12CCC2 42353,C1(NC(C2CCc3nn[nH]c3C2)=O)CC1C1CCCN(C(C2CC2F)=O)C1 42354,c1(NC(c2nnc3ccccn23)CCC)nccc(=NCCCNC(C)(C)C)[nH]1 42355,C1(C(N(C2CCN(C(c3ncc(F)cn3)=O)CC2)CC#C)=O)CN(C)CC(C)O1 42356,CN1CC(O)CC1C(=O)NCCN(CCOCCO)C(C1C(CO)C1(F)F)=O 42357,C1(C2(O)CCN(C(c3ccsc3Cl)=O)CC2)(Nc2cc3nnc(C)n3cn2)CC1 42358,C1(c2ncc(C)s2)CCCCN1CC#CC(C)(C)C 42359,C1(NC(c2coc3c2CCCC3)=O)Cc2ccccc2N(C(c2ccns2)=O)C1 42360,c1(C(=O)NCCC2(O)CCCN(C(C(CC)(C)C)=O)C2)cc(O)cc(F)c1F 42361,N1(C(C(C)OCOC)=O)CCC(C(=O)NCCc2cnnn2C)C(C)(C)C1 42362,N1(C(c2cc(F)c(F)cc2F)C(=O)NCC(F)F)CCc2cccc(Br)c2C1 42363,C1(NC(C2=NNC(=O)C2)=O)CCCCN(C(c2ccnn2CC(F)(F)F)=O)CC1 42364,C1(NC(C2(C)N(C(c3cc(C)no3)=O)CCC2)=O)CCCN(CC(F)(F)F)C1=O 42365,c1(C(N2CCC(NC(CC3C(C)C3)=O)C(C)(C)C2)=O)n[nH]c2ccc(F)cc12 42366,c1(NC(C2CCCC(NC(C3CC(O)C3)=O)C2)=O)ccc(Br)c(Cl)c1 42367,c1(CC)nn(C)cc1C(=O)NC(C)(C)CC(=O)NCC(O)C(F)(F)F 42368,CCC(C)(CCC(C)C)C(=O)N1CCC(N(CCO)C(C2CCNC(=O)C2)=O)C1 42369,c1(C(=O)NC2CC(CNC(C3C(CC)OCC3)=O)C2)cc(C)cc2c[nH]nc12 42370,C1(NC(c2n(C(C)C)ncc2)=O)C2CCC1CN(C(c1ccc(F)cc1Br)=O)C2 42371,c1(C(=O)NCCCC(C)(C)NC(C=CCC)=O)ccc2c(c1)C(=O)NC2=O 42372,Cc1cc(C(N2CCCC2CCNC(=O)CS(=O)(=O)N(C)C)=O)nc(O)n1 42373,CC(CC(=O)NC1CCCC1NC(C1(C(F)F)CC1)=O)n1cccn1 42374,O=C(CC1CC2CC1C2)NNc1ccc(Br)c(F)c1F 42375,Cc1ccc(OCC(N2CCC(CNC(C34CC(CF)(CO3)C4)=O)C2)=O)c(C)c1 42376,Cc1cc2[nH]c(C(=O)Nc3ccc(C4CCCN(c5ccncn5)C4)cc3)cc2s1 42377,c1(N2CC(NC(C=C(C)Cl)=O)CC3(C2)CC3)nc2cc(F)ccc2o1 42378,c1(CSCCC)ccc(NC(=O)NC2(O)CCCSC2)cc1 42379,CCCC(CC)C(=O)NCC1(C)CCN(C(C2(CC3CC3)CCOCC2)=O)CC1 42380,C(=O)(C(F)C(F)(F)F)NC(CC)CNC(=O)COCc1ccncc1 42381,CC1(C)CC(NC(=O)C(C)(F)C(C)(C)F)CCN(C(c2c(O)cccc2F)=O)C1 42382,Cc1nc(C(=O)NCC2(C)CCN(C(=O)Cc3cnc(C)s3)C2)c2ccnc-2[nH]1 42383,c1(N2CCN(C(=O)Nc3cccc(F)c3)C3C2C3)ncnc2sccc12 42384,C1(C(=O)NCC(CC)OC)CN(C(c2ccccc2N(C)C)=O)CCC1O 42385,C12(C(N(C)CC3N(C(C4C(CC)N(C)CC4)=O)CCCC3)=O)CCC(CC1)OC2 42386,c1(C(=O)NC2CC(CNC(C(CCC)C)=O)C2)ccc2nc(O)cn2c1 42387,c1(C(N(C)CC2N(C(C(C)(CO)OC)=O)CCC2)=O)cc2c(cn1)COCC2 42388,c12cc(OC)c(c(Cc3cnc[nH]3)c1)CN1CC3CC(C1)N23.CO 42389,C1(C(=O)NC(C2(O)CCN(C(c3cnsc3)=O)C2)C)CCN(C)C(=O)C1 42390,CC(C(=O)NCC1(F)CN(C(c2ccc(SC(F)(F)F)s2)=O)C1)S(N)(=O)=O 42391,c1(N(C)C)cccc2sc(C(N3CCC3CNC(=O)CSCC(N)=O)=O)cc12 42392,N1(C(CC2CC(=O)C2)=O)C2CCCC1CC(NC(C13CSC(C1)C3)=O)C2 42393,c1(C(=O)NCCN(C(=O)CN2CCC(C)C2)CCOC)nccc(Br)c1C 42394,C1(NC(CNC(C(c2ccccc2)C)=O)=O)CC(C)(C)C12CC2 42395,CCCCC(O)CC(=O)NC1CCCC(NC(=O)COc2c(F)cccc2F)C1 42396,C1(CCNC(CCC#C)=O)CC(F)(F)CN1C(=O)C=Cc1scnc1C 42397,C(CCCCCNC(c1sc(COC)nc1C)=O)NC(c1c(CCC)[nH]cc1)=O 42398,N1(C(C2CCC(CC)CC2)=O)CC(C)N(C(c2nnn3c2CSCC3)=O)CC1C 42399,C(=O)(C#CC1CCCCC1)NC1CC(C(=O)NC(CC=C)CC(F)F)C12CCC2 42400,C1(NC(C=CC=CC)=O)CCC12CN(C(C1(CC(=O)OCC)CC1)=O)C2 42401,C1(C(=O)NCc2c(C(=O)NCCCn3cccn3)nco2)(CC)CCCC1O 42402,n1(CCC)ccc(C(=O)NC2CCC2CNC(C2CNC(=O)N2)=O)n1 42403,Cc1ccc(C(=O)NC2(C(=O)NCc3ccc(CO)o3)CCCC2)c(O)n1 42404,C1(NC(=O)C(=CC2CCCCC2)F)CCN(C(=O)C(N2CCCC2)C2CC2)C12CC2 42405,NS(=O)(=O)C1CN(C(=O)NCNC2COCCC2(F)F)C2(CCC2)C1 42406,CC1CC2CN(C(c3cnc4[nH]cncc3-4)=O)CC2N1C(=O)CCCS(C)(=O)=O 42407,C1(C)(C(c2n(CC(=C)C)nnn2)NCCc2cnoc2)CCCC(F)(F)C1 42408,c1(N(S(=O)(=O)C(Cl)(Cl)Cl)CCC)cccc(-c2cscc2CO)c1 42409,c1(CN2CCN(CC(=O)Nc3ccc(OC)c(O)c3)CC2)c(F)cc(Br)cc1F 42410,c1(C(=O)NCCC2CCN(C(C(CC#C)(C)C)=O)C2)ccc2c(O)n[nH]c2c1 42411,C(CC(=O)N1CCOC(CC)CC1)(C(F)(F)F)NC(C(CCCC)N(C)C)=O 42412,c1(OC)cccc(OC)c1S(=O)(=O)Nc1nc(C)cs1.C12C3CN(CC13)C2=O 42413,C1(N(C(=O)C(c2ccnn2C)OC)CC)CCN(C(=O)CNC(=O)C2CC2)CC1 42414,C(=O)(CCCC(F)(F)CO)NCCOCCCNC(C1C(C)OC(=O)N1)=O 42415,CCC(C)(C(=O)NCC1CC(NC(c2cnccc2C(C)(C)C)=O)C1)OC 42416,c1(CC)cc(C(=O)NC2CC23CCN(C(=O)CCC2CC(OC)C2)C3)ccc1F 42417,Cc1ccc(CC2(CC(N3CCN(C(C4CCCS4(=O)=O)=O)CC3)=O)CC2)cc1 42418,c1(OC)ccc(CN2CCN(C(C3CC3C)=O)C(C)C2)nc1Cl 42419,c1(CC(N2CC(NC(c3csnn3)=O)CC(C)C2)=O)cccc2ccoc12 42420,C1(CC(=O)NC2CC=C(C)CC2)N(C(c2csc(F)c2)=O)CCC1(C)C 42421,N1(C(CC2C(C)(C)COCC2)=O)Cc2cccc(CNC(c3ccns3)=O)c2C1 42422,Cc1c(CN2CCC(SC(C)(C)C)C2)occc1=O 42423,C(=O)(C(c1cccs1)NC(=O)C(C)N1CC(C)C1)NCC(=O)OCC 42424,N1(C(C(C)NC(=O)OC)=O)CCCC(NC(c2cccc(C(F)F)n2)=O)C1 42425,C1(NC(C2C(C)CCN2C(C2C3CCCC23)=O)=O)CC2(C1)CC(C)(C)C2 42426,C(C(F)(C(=O)NC(COCC1CC1)CC)C(C)C)NC(c1c(CC)nco1)=O 42427,c1(C(=O)NCC(C2CCC2)NC(c2c(C(C)(C)C)ncs2)=O)cc[n+]([O-])cc1 42428,N1(C(c2cnn(CC)c2Br)=O)CCC(NC(=O)Cn2ccc(C)n2)CC1C 42429,C12(NC(C3(OCC)CC3)=O)COCC1CN(C(=O)C(C1CCC1)OCC)C2 42430,C(CCCCCN(C)C)NC(C(C1CCCO1)NC(c1c(C)occ1)=O)=O 42431,c1(C(=O)NCC(C2CCOC2)NC(c2ccon2)=O)snnc1-c1ccccc1 42432,C(=O)(C(C)(C)C(C)C)NC(CN(C(c1sc(-c2ccsc2)nc1C)=O)CC)C 42433,c1(C(N(C2CCN(C(C(Br)=C(C)C)=O)C2)CCO)=O)cnn2c(N)ccnc12 42434,C1(C(=O)OC)CC1C1CCN(C(=O)Nc2cccc(NC(C)=O)c2)C1 42435,C(=O)(C(O)CCCNC(c1cnnn1C1CC1)=O)N(C)CCOC(F)F 42436,N1(C(c2c(C)cc[nH]2)=O)CC(C)C(NC(c2cnc(C(C)(C)C)[nH]2)=O)C(C)C1 42437,N1(C(c2n(C)nc(O)c2)=O)CCCC(CNC(c2c[nH]c(Br)c2)=O)CC1 42438,c1(-c2nnc(N(CCC)C)n2CC(=O)N(C)C)cc(Cl)ccc1OCC 42439,Cc1c(C(N2CC3CC(C2)N(C(=O)C(C)C#N)C3)=O)cc(Br)cc1Cl 42440,N1(C(C(CCC#C)O)=O)CCCN(C(=O)CCCc2cccs2)CC1CO 42441,C(=O)(C1=CC2(CCOC2)C1)NC1(C2N(C(c3c(C)nc(O)[nH]3)=O)CCC2)CC1 42442,C(=O)(C1=CCCOCC1)N1CCCC(CC=C)(NC(=O)Cc2cnn(C)c2C)C1 42443,c1(-c2cncc(OC)c2)cc(C)cc(F)c1 42444,C=CC1(CC(=O)N(CCO)CC2CC2)CN(C(=O)C(C)(C)n2cncn2)C1 42445,C1(CC)CN(C(c2cc(Cl)cnc2C)=O)CCN1C(c1ccc(C)o1)=O 42446,Cn1nc(C2CC2)cc1C(=O)Nc1cccc(NC(c2cc(C3CC3)no2)=O)c1 42447,CC(CC1CC1)C(=O)N(CCCOCCNC(C1(C2CCCO2)CCC1)=O)C 42448,N1(C(C(N(C(=O)CCCc2ncco2)C)C2CC2)=O)CCC12CCCC2 42449,N1(C(c2n(C)nc(O)c2)=O)CCC2(CCC2CNC(=O)COC2CCCC2)CC1 42450,C1(NC(c2scc(C(=O)OC)n2)=O)Cc2ccccc2C1C#N 42451,Cc1cc(C)c2cc(C(N3CC(F)CC3CN(C(=O)C(C)N(C)C)C)=O)sc2n1 42452,C=CC(C)(CCOC)C(=O)NC(CNC(=O)C(C)C(=O)OCC)CO 42453,c1(OC)cc(F)c(C(=O)NCC2CC(C)N(C(C3CC(=C(C)C)C3)=O)C2)cc1N 42454,C1(C)(C(N2CCCC(N(C(=O)CSC(C)C)CC)C2)=O)CCC(C)C1(C)C 42455,c1(C(=O)NC(CCC)CNC(=O)C(F)Cc2ccccc2)nccc(C)c1N 42456,C1(NC(CC2CCCC(OC)C2)=O)CC(C)CN(C(=O)C=CCO)C1 42457,O=C1CC2CC(C(=O)NCC3OCCC3C(=O)NOC3CCC3)C1O2 42458,Cc1nc(O)nc(O)c1CCC(N1CCN(c2ccc(C#N)nn2)CC(O)C1)=O 42459,c1(CC)cc(C)c(C(=O)NC2CC(CCn3cc(CC4CCCOC4)nn3)C2)o1 42460,Cc1nocc1CC(=O)N(CCCNC(C1CCCN1C(=O)NC1CC1)=O)C(C)C 42461,Cc1c(C(N2CCC(C(C)(C)CNC(=O)C(C)(C)C3CCCO3)CC2)=O)nnn1C 42462,C(=O)(C(C(C)(C)C)n1ccnn1)NC1CCC(NC(c2nn(CC)nc2C)=O)C1 42463,C1(NC(C(C)=C(C)C)=O)CCN(C(=O)CCOCC2CC2)CC12CCC2 42464,S(=O)(=O)(c1cccnc1NCC1=CCCOC1)NC(CC)CSC 42465,c1(CC)ccc(F)c(C(=O)NCC2CN(C(=O)Cc3cscn3)CCCO2)c1F 42466,C(c1ccccc1Br)=CC(N1CC2CC2(C(N2CCCCC2CCO)=O)C1)=O 42467,C(CC1=CCN(C(C23CC(C(=O)OC)(CO2)C3)=O)CC1)NC(C(C(=C)Cl)(C)C)=O 42468,C(=O)(C(C)C(C)NC(=O)C(N)=O)N(CC=C)C(C)C 42469,C1(C)(C(N(CCC(=O)NC2CCN(CCOC)C2)C)=O)CCC(=O)N1 42470,c1(C(N(CCN(C(c2nnn(C)n2)=O)CC)CC)=O)cc([N+](=O)[O-])n[nH]1 42471,C1(C(=O)NCC2CC(OC)CN2C(=O)COC2CCC2)C2CCC1(C)C2(C)C 42472,c1(C(N2CC(SC)C(NC(=O)C(F)n3ccnc3)C2)=O)cc(C)cc(C)c1 42473,N1(C(COCCC)=O)CC2CC(NC(C3(C(C)C)COC3)=O)C(C2)C1 42474,N1(C(C(N2CCOC2=O)C)=O)CCOCC1CC(N1CCCC(F)C1)=O 42475,CCC(CC(=O)N1CCN(C)C(C(=O)NCC2(C)CC(C)C2)C1)C(C)(C)C 42476,c1(C(N2CCCC(Cn3cc(C(CC)(C)O)nn3)C2)=O)c(C)[nH]c2ncccc12 42477,C1(C(=O)NCC(C=C)O)CC2CC1CN(C(=O)CC=CCC)C2 42478,CC1CN(C(c2csc(F)c2)=O)C(C)CN1C(c1ccnn1CCF)=O 42479,CCCC(CNC(=O)C=CC1CCOCC1)C(=O)N1CCC(c2cnn[nH]2)C1 42480,C1(CNC(c2c(OC)cnnc2)=O)CC(C)CN(C(=O)Cn2nc(C)cc2C)C1 42481,N1(CC(=O)NC(C(=O)NCCC(=O)OC)(C)C)CCC(F)CC1 42482,CCC(C)(C)CCNC(=O)CC1CCC(NC(=O)CC2(OC)CCC2)C1 42483,CN1CCCC(CCC(=O)NC2(CNC(C3CSCCS3)=O)CC2)C1 42484,C(=O)(CCCCCCCSC)NC1C(NC(c2cccc(CC)n2)=O)CCC1 42485,N1(C(C2(OC(C)=O)CC2)=O)CCC2(CC1)CC(C)N(C(=O)CCC1CCCO1)C2 42486,c1(COCC(=O)NC2CC(C)(NC(C3CCCCO3)=O)C2)cccc(C(F)F)c1 42487,N1(C(c2c(=O)ccn(C)c2)=O)CC2CCC(C1)C2CNC(c1ccn(C)c1)=O 42488,c1(CN(C)Cc2ncn(C)n2)cc(F)ccc1CN1CCCCC1 42489,N1(C(C=CCOC)=O)CC(C)(NC(=O)COCC2CCCO2)C1 42490,c1(C(=O)NC(C(C)NC(CCc2c(C)ncs2)=O)CO)ccn2ccccc12 42491,C1(C2(O)CN(C(C3CC3CC(C)(C)C)=O)C2)(CNC(C2CN(C)C(=O)C2)=O)CC1 42492,C#Cc1cccc(CC(=O)NC2CN(C(C3COCC3C(N)=O)=O)CC2OC)c1 42493,N1(C(c2c(C)nc(O)cc2)=O)CC2(C(=O)NC(C)C(F)F)CC1CCO2 42494,C1(C(=O)Nc2c(C(=O)OCC)cno2)CC2CC2N1C(c1cc(O)ncn1)=O 42495,N1(CC)CCC(C(=O)NC2CCC(C(=O)N(C3CC4CC4C3)C)C2)C1 42496,CC#CCCC(=O)NC(c1ccccc1)CNC(c1[nH]cnc1C)=O 42497,C(=O)(C(C)C(O)CCCC)NCC1CCC(N(C(CCCCC#C)=O)C)CC1 42498,n1(CC)nc(C)cc1C(N1CC2C(C1)N2C(=O)Cc1csc(C)n1)=O 42499,Cc1ccc(CC(=O)NCC(O)CCNC(C2(N3CCOCC3=O)CC2)=O)cc1 42500,C1(C(=O)NC(CC(=O)N(C2CCN(CC)CC2)C)(C)C)CC2(CCCO2)C1 42501,C1(C(=O)OC)C(F)(F)C12CC(C(=O)NC(C)(CNC(c1cc[nH]n1)=O)CO)C2 42502,c1(C(N(CC(CC)NC(c2n[nH]c(C)c2Cl)=O)CC)=O)ccc2nnnn2c1 42503,c1(-n2c(C3CCOCC3)nc(-c3scc(C)n3)n2)c(C)cc(C)cc1C 42504,C1(N(C(c2cscc2OC)=O)CC)CCCN(C(=O)C(C)=CC(C)(C)C)C1 42505,S(=O)(=O)(c1ccc(C#N)cc1Cl)N1CCC(N(C)Cc2cc(Br)c(Br)s2)C1 42506,C(=O)(C(CC)C(C)O)N(C1CCC(NC(c2c(CC)nco2)=O)CC1)C 42507,c1(CNC(=NCCOCC)NCc2ccoc2)nn(C)c(C)c1S(N)(=O)=O 42508,C1(C(=O)NCC2C(C)(C)COC2)CCC2(CC2)N1C(c1cc(C2CC2)no1)=O 42509,N1(C(=O)COC2CC2)CCC2(CCN(C(c3cc(Cl)c[nH]3)=O)C2)C1 42510,n1(CC)c(C(N2CC(C)C2C(=O)N(C2CN(C(C)C)C2)C)=O)cnc1O 42511,C1(C(=O)NC(C(=O)Nc2csc(Cl)c2)c2cccs2)CC1C1CCC1 42512,c1(NCc2cnc(CC)[nH]c2=N)cc(=NC2CCCN(C)C2)[nH]c(CC)n1 42513,N1(C(c2c(C)nccc2)=O)CCC(C)C(NC(=O)CC2CCCC(F)(F)C2)C1 42514,n1(COCC)nnc(C(=O)NC2CCN(C(=O)COC(F)F)CC2)c1N 42515,C(=O)(C#CC1CCCO1)N1CC(CNC(Cc2[nH]c(=N)sc2)=O)C(C(F)(F)F)C1 42516,Cc1ncn(C)c(=O)c1C(=O)NCCN(C(=O)CNC(C1CCC1)=O)C 42517,C(=O)(C(CC(C)(C)C)OC)N1C(CC=C)(C(=O)NC(CCF)C(=O)OC)CCC1 42518,N1(C(C(C)C(C)(C)C)=O)CC(NC(=O)CN2CCCNC2=O)C(S(C)(=O)=O)C1 42519,Cc1nn(C)cc1NC(C1C2CC2CN1C(C1CCC1C#N)=O)=O 42520,c1(C(=O)NC2(CC)CN(C(CSCC)=O)C2)cc(NC)nc(Cl)c1 42521,c1(CNC(C(CNC(C2CCCN2C)=O)OC)=O)cnccc1Cl 42522,CCC(C)C(C)C(=O)N1CCCC(CNC(c2c(Cl)n[nH]c2C2CC2)=O)C1 42523,C(=O)(C(CN(C)C)NC(C1CCCN1C1CC1)=O)N(CCNC(C)=O)C 42524,C1(C(N2C3C(NC(CC4CCN(C)C4)=O)C(CC3)C2)=O)CC(C)(C)CC(C)(C)C1 42525,Cc1cnccc1C(C)C(=O)NCC(C)(O)CNC(=O)CCc1cccnc1 42526,CCN=C(NCc1nccn1CCc1ccco1)N1CCOC(C(F)(F)F)C1 42527,C1(NC(c2on(C)c(=O)c2)=O)CCN(C(=O)CCOc2cccc(Cl)c2)CC1F 42528,C(=O)(C(CCSC)N(C)C)N1CC(NC(C2C(CC)OCC2)=O)(CO)C1 42529,c1(-c2c(F)ccc(SCc3n(C)ccn3)c2)cccc2c(CC(=O)O)cccc12 42530,N1(C(CSS(C)(=O)=O)=O)CCC2CN(C(=O)COCC3CCCO3)CC12 42531,c1(SC)nc(=N)[nH]c(=NC(C)C2CCCN(C(C3C(C4CC4)C3(F)F)=O)C2)[nH]1 42532,C#CC1CCCCN1C(C1(C#C)CN(C(=O)CC23CCC(CC2)C3)C1)=O 42533,C=C(Br)CN=C(NCc1ccco1)NC1CCC1C 42534,c1(N(C)C)cccc(-c2cnc(C(=O)N(CCN(C)C)Cc3nccn3C)[nH]2)c1 42535,C1(CCN(C(CCN(C)CC)=O)C)CCCCN1C(c1csc(Cl)n1)=O 42536,c1(C(=O)NCC2(CNC(c3c(OC)c(=O)cco3)=O)CC2)nc[nH]c2ncnc1-2 42537,CC(=O)CCCCCCC(=O)N1CCN(C(C2CC3CC3C2)=O)CCC1C 42538,CC12COCC1CN(C(=O)C(c1cccnc1)NC(c1cnc(O)o1)=O)C2 42539,N1(CC)C(=O)CCC1C(=O)N(C(C)CCNC(=O)CC1CCCCO1)C 42540,C1(CC(=O)NC)CN(C(=O)CCCN(C)C)CCN1C(c1cccc(=O)n1C)=O 42541,C1(NC(CCC=CC(C)C)=O)CC2C1CCN2C(=O)CC(C1CCC1)C1CCC1 42542,N1(C(C(CC)N(C)C)=O)CC2(CCN(C(=O)Cn3ncnn3)CC2)C2COCC12 42543,C1(C)(C(N2CCC(N(C(=O)Cc3nnc(-c4ccco4)o3)C)C2)=O)CCC(O)CC1 42544,C1(C(N(CCCC)C2CC2)=O)CN(C(C2CC23CCCC3)=O)CC1C1CC1 42545,Cc1nsc(C)c1C(=O)NCc1cc(C(N2CCCC2CC2CCC2)=O)n[nH]1 42546,C(c1cc(F)cc(F)c1)=CC(N1CCN(C(C2CC2F)=O)C(CC2CC2)C1)=O 42547,CN1CC(CCNC(=O)CN(C)C(c2ccc(C3CC3)o2)=O)CC1=O 42548,C1(C)(CC)C=C(C(=O)NCC2(C)CCN(C(c3c[nH]nc3F)=O)CC2)C1 42549,c1(C(=O)NCC(C)(C2CCC2)NC(CN(C(=O)OC)C)=O)cc2ccnn2cn1 42550,c1(OC)cc(CNC(C2CC2NC2CC2)=O)cc(F)c1OC.C(CC(C)C)S 42551,N1(C(C2(C=C)CCC2)=O)CCCCC1C(C)NC(=O)CCCCNC(N)=O 42552,C1(C(=O)NC(CCN(C(C2(NC(C)=O)CCCC2)=O)C)C)CCS(=O)(=O)C1 42553,C=C=CC(C)C(=O)NCCOCCOCCNC(C1(C#N)CC(C)C1)=O 42554,N1(C(C(=O)NC(CC)CN(C(=O)Cc2nc[nH]n2)CC)C)CCCCCC1=O 42555,c1(C2(C)CC(NC(C(c3ccccc3F)OC)=O)C2)cccc(Cl)c1 42556,c1c(F)cccc1F.N(C(=NCC1CC1)NCc1ccnn1C)Cc1nnn(C)n1 42557,C1(CC)CCCCC1OCC(=O)NC(C1CCN(C(=O)C(=O)NC)C1)C 42558,C12(OC)CCC1CN(C(C13CC(CO1)N(C(=O)CCc1cnccn1)C3)=O)C2 42559,c1(CNC(C2CN(C)C2)=O)ccc(C#N)cc1.CC1C2CCN1C2=O 42560,C1(C(=O)NC(C(=O)NC2CCOCC2)c2ccco2)Cc2nccn2C1 42561,n1(CC(=O)Nc2c(C)cc(C(F)(F)F)cc2)nc(CN)c2c1CCC2 42562,c1(C(=O)NCC2CCN2C(C23CC(CO2)C3)=O)nc(Br)c2ccccn12 42563,C1(NC(c2cccc(C#C)c2)=O)CN(C(=O)C(C)SC(F)(F)F)CC12CCC2 42564,c1(C(=O)NC2C(NC(c3nc(OC)c(F)cn3)=O)CCC2)c(F)cc(N)cc1F 42565,N1(C(C2(NC(C(COC)C)=O)CCC2)=O)CC(O)(C2CCC2)C1 42566,N1(C(C(C2CCCCC2)C)=O)CCC(CNC(=O)C(O)C2CC2)C1(C)C 42567,C=C1c2ccccc2C(=O)N1CC(N1CC2(C1)CN(C(C1NC(=O)OC1C)=O)C2)=O 42568,Cc1cccc2c(CC(N3CC4CC4(NC(c4c(Cl)cnn4C)=O)C3)=O)c[nH]c12 42569,N1(C(Cc2c(C)nn(C)c2)=O)CC2(CC(C(=O)NOCCOCCO)C2)C1 42570,c1(C(=O)NC(c2ccccc2)C(C)NC(CC(=C=C)C)=O)cc(C)ccc1F 42571,c1(C(N2C(CNC(C(CC)(C)CO)=O)CCCCC2)=O)onc2ccccc12 42572,N1(C(CC(=O)N(C)C)=O)CCC(CCC(=O)N(C)Cc2nccn2C(C)C)CC1 42573,C1(C(=O)NC2(CN(C(=O)C(C)(C)c3ccn(C)n3)C)CC2)CCCCCC1(F)F 42574,CCCC(CC1CCCC1)C(=O)N1CCC(O)(CNC(c2[nH]nnc2C)=O)CC1 42575,CC12CCN(CC1)CC2C(=O)NCC1CCN(C(c2c(F)ccc(F)c2N)=O)C1 42576,C1(S(C)(=O)=O)(C(=O)NCC(CO)NC(Cc2c(C)ccc(C)c2)=O)CC(O)C1 42577,N1(CCCNC(=O)NCc2cncc(C(=O)OC(C)(C)C)c2)CCCCS1(=O)=O 42578,N1(C(c2ncoc2C2CC2)=O)CCC2CC2(C(=O)NC2(CO)CCC2)CC1 42579,c1(C(C)N(CCN2CCCC2)C2CC2)cccc(C2CCCC2)c1 42580,N1(C(COCCC=C)=O)CCC(C)(CCNC(c2ccc(OCCF)cc2)=O)C1 42581,C1(NC(CSCCC)=O)CCCN(C(=O)C(c2ccc(OCC)cc2)C)CC1 42582,C(=O)(CC(C(F)F)c1ccccc1)N(CCCN(C(C=CC=CC)=O)C)C 42583,c1(COC)nc(N2CCCC(N(C(=O)CC3(O)CCC3)C)CC2)cc(Cl)n1 42584,N1(C(C(F)=CCC)=O)CC(C)CCC1CNC(=O)COC1(C)CCC1 42585,c1(C(=O)NC(CC=C)CNC(c2c(Cl)sc(Cl)c2C)=O)cccc2nonc12 42586,c1(CN(CCN(C(C2(NC)CCSC2)=O)C(C)C)C)ccc(C)c2cccnc12 42587,c1(CN2C(C(C3CC3)NC(c3cccc(OC)n3)=O)CCC2)cccc(F)c1Cl 42588,c1(C(N(CCN(C(=O)C(F)C(C)C)CC)CC)=O)ccc2c(c1)COCCN2 42589,C=CC1(C(N2CC(CCNC(C3(CCF)CC3)=O)C2)=O)CCCCC1 42590,COn1cnc(C)c1C(=O)NCCCN(C)C(c1sc(Br)cc1C)=O 42591,C1(CC(=O)N(CC(=O)NC(C)CN(C)C)C)(NC(C)=O)CC1 42592,c1(C(=O)NC(CC)(CNC(C2(CO)CC2(F)F)=O)CC)cnc2c[nH]nc2c1 42593,Cc1nc(C(C)C)sc1C(=O)N(CCN(C(=O)COc1ccsc1)C)C(C)C 42594,c1(CC(=O)NCCCN(C(=O)C(O)C2CCC2)C2CC2)csc(C2CC2)n1.O=CN 42595,N1(C(C2(C(N(C)C)=O)CC2)=O)C2CCC1CC(NC(C1CC13CC3)=O)C2 42596,C1(C(N(CCO)CC)=O)CCOC1CNC(C1C=C(C)CS1)=O 42597,Cc1ncc(C(N2CCC(CCNC(=O)C(F)C(F)(F)F)CC2)=O)cc1N 42598,Cc1cc(C(=O)NC2CC(O)CN(C(=O)COc3cccnc3)C2)c(F)cc1N 42599,c1(C(=O)NC2C(CC)N(C(C3CCOCC3)=O)CCC2)cc(F)c(C)cc1N 42600,C12(CNC(c3ccc(CC)nc3)=O)CCCC1CN(C(C1CC(C3CC3)C1)=O)C2 42601,n1(CC(=O)NCC2N(C(CCCC=C)=O)CC(F)C2)nc2n(c1=O)CCCCC2 42602,C(C(=O)NC(C)C(C)NC(=O)C(c1ccc(F)cc1)(C)C)(C(C)C)NC(C)=O 42603,C(=O)(C(CCSC)N(C)C)N(C1CCC(NC(=O)CC2(OC)CCC2)CC1)CC 42604,N1(C(C=COCC)=O)CCC(n2cccn2)(CNC(C2CC2C(F)F)=O)CC1 42605,CC1(NC(C2CCC(P(C)(C)=O)C2)=O)CCCc2ccccc21 42606,c1(COC)ccc(C(=O)NCCCC(C)NC(=O)CC2CCC(=O)N2C)cc1 42607,Cc1cc(O)cc(=O)n1C(C)C(=O)NCCC1CCCN1C(=O)CN(C)C(C)C 42608,C(CC(=O)NCC1CCOC1=O)(CC(C)C)NC(CSCC#C)=O 42609,CCC(CC(=O)NCCCC(C)(C)NC(=O)C(CO)C(C)(C)C)C(C)(C)C 42610,C1(OC)(OC)CC(C)(CNC(c2cnn(CCO)c2C2CC2)=O)C1 42611,N1(C(CN2CCN(C)CC2)=O)CCC2CN(C(=O)C(C)(O)C3CCCCC3)CC12 42612,c1(C(N2C(C)(CNC(C(C=C)(C)C)=O)CCC2)=O)cccc2oc(C)nc12 42613,Cc1ccccc1COCC(=O)NC1C2CC1N(C(C1(C)CC(C)C1)=O)C2 42614,N1(C(C2(OC)CCC2)=O)CCC2C(CCN2C(c2cc(C)ncc2Cl)=O)C1 42615,Cc1cc(C(N2CC(C(=O)NCCSC(F)F)CCC2C)=O)nnc1C 42616,Cc1c(C(=O)NC2C=CCC(C(N3Cc4c[nH]nc4C3)=O)C2)cccc1F 42617,c1(CC)cc(N2CC3CC(NC(C4CCCC4CC)=O)C3C2)nc(CC)n1 42618,N1(C(c2cc(CC)n(C)n2)=O)CCCC(N(C(=O)Cc2ccc(Cl)cn2)C)CC1 42619,C(=O)(N=c1cc(C)n(-c2ccccc2Cl)[nH]1)Nc1n(CCCC)ncc1 42620,c1(CN2CC3C(CNC(c4cc(C(F)F)no4)=O)C3C2)ccc2ncnn2c1 42621,CCCCC(CNC(=O)C(CC)OC1CCCC1)NC(C1CC(F)C(=O)N1)=O 42622,c1(C(N2CC(O)(C(C)NC(C(CSC)C)=O)C2)=O)ccn2cccc2c1 42623,N(C1CN(C(=O)C(O)CC2CC2)Cc2ccccc21)C(c1c(C)nc[nH]1)=O 42624,C1(NC(C2CC(CCC)C2)=O)CCCC(C(N2CCSCC2)=O)CC1 42625,N1(C(C(N2CCC(O)CC2)C)=O)CCC2(CC1)CC(=O)NC(=O)N2 42626,C1(NC(c2ccc(CO)cc2F)=O)CCN(C(=O)CSC(F)(F)F)CCC1(F)F 42627,N(C1CN(C(=O)CC2(C)CC2)Cc2ccccc21)C(c1cc(C)no1)=O 42628,C1(c2cn(CCNC(c3ccncc3F)=O)nn2)CC2CCC1O2 42629,c1(C(=O)NC(C(C)NC(CCC(=O)NCCC)=O)C)cc(C)c(C)nc1C 42630,c1(C(=O)NCC2(COC)CC2)c(NC(CO)=O)cccc1F.C(COCC)OC 42631,CC1CN(C(=O)Cc2n[nH]cc2Br)CCC1N(C(=O)CSCC(N)=O)C 42632,C1(N(C(C=CC(CC)=CC)=O)CC)CCCN(C(c2ccncc2CC)=O)C1 42633,CC1CC(C)(C(N2CC(CCCCNC(c3csc(Cl)c3Cl)=O)C2)=O)CC(C)O1 42634,CC(C)(C(=O)NCCC1CN(C(=O)COc2ccsc2Cl)C1)C(F)F 42635,c1(C(=O)NCC(=O)NCC(=O)NCc2nc(C)sc2)ccnnc1O 42636,c1(OC)ccc(C(N2CCC(CNC(=O)CC(C)OC)(OC)C2)=O)cc1F 42637,c1(NC(C(C)OCC)=O)cccc(NC(c2snnc2C(C)C)=O)c1 42638,N1(C(CC(C)(C)OC)=O)C2CCC1CN(C(c1cnoc1C)=O)CC2 42639,C1(CNC(C=CC(C)C)=O)CC(NC(c2coc(C3CCOCC3)n2)=O)C1(C)C 42640,C(=O)(C(C)CC(N)=O)NC1(C)CCN(C(Cc2cccc(C)c2)=O)C1 42641,N1(C(C(C)n2cccc2)=O)CC2CC1CC2CNC(=O)C(C)(C)c1cnn(C)c1 42642,c1(C(=O)NCC2(CNC(c3ccc(C)nc3)=O)CCCC2)cc(F)cnc1O 42643,N1(C(CC2C(C)=NNC2=O)=O)CC2CCOC2(CNC(=O)CCc2c[nH]cn2)C1 42644,c1(OC)cc(C)nc(N(C)CC2CCN(C(=O)CC(C)SC)CC2)n1 42645,C1(CC)C(C(=O)NCc2nc(CO)n[nH]2)CCN1C(=O)C(c1cncnc1)C 42646,C1(c2n(CC(=C)C)nnn2)(NCc2cc(Br)no2)CCC2(CCOCC2)C1 42647,Cc1cccc2cc(C(=O)NC3(CNC(C45CC(F)(C4)C5)=O)CCOC3)nn12 42648,c1(C(=O)OCC)n[nH]c2c1CCC(NC(C)Cc1ccc(O)cc1)C2 42649,c1(NC)ccccc1C(N1CCC(C)(CNC(=O)CCc2ccnc(Cl)c2)C1)=O 42650,CC(F)(F)CC(=O)N1CCN(C(=O)CCc2cnccn2)CC1 42651,c1(N2CC(C)(NC(CC)=O)C2)nc(C(F)(F)F)ccc1C(=O)OCC 42652,CCC(C)C(O)C(=O)NC1CC(CCNC(=O)C(F)C(F)(F)F)C1 42653,C1(N(C2CC3CC2CN3)C(=O)COCCOC)CCNCCC1C 42654,S(=O)(=O)(c1ccc(N2CC(C)C(O)C(C)C2)nc1)NCC(=C)CC 42655,N1(C(c2ncn(C)c2)=O)CC2CCC(C1)N2C(=O)Cc1cnn2ccccc12 42656,C1(C)(N(C(=O)COc2ccn(C)n2)C)CCN(C(=O)CCc2cccs2)C1 42657,c1(C(=O)NCCC2(CNC(C(CC#C)C)=O)CC2)ccc2c(Br)n[nH]c2c1 42658,C#CC1(O)CCN(C(C2(C)CCN(C(=O)C(O)CC(C)(C)C)C2)=O)CC1 42659,C1(CC(=O)NCCc2cc(C)ncc2)N(C(=O)C=Cc2ccco2)CCC1(C)C 42660,C1(NC(c2n(C)nnn2)c2ncc(-c3ccccc3)s2)C(=O)OC2CCCC12 42661,C(C)(C)(CC(C)NC(C1(NC(=O)C=Cc2ccc(C)o2)CCCC1C)=O)OC 42662,c1(OCC)n[nH]c(C(=O)NC2CCCC2c2nc[nH]n2)c1Cl.c12c(cnn1C)SC2 42663,CCC1=C(C(=O)N2CCCC2CN(C)C(c2c(Br)noc2C)=O)CCCO1 42664,c1(C(=O)NCC(C)NC(c2csc(-n3cccc3)n2)=O)ccc(N(C)C)cc1 42665,N1(C(C(CC)N(C)C)=O)CCC2(C=C(C(=O)NCCc3ccc(C)cn3)C2)C1 42666,C(C(=O)N=c1ccn(CCO)[nH]1)(c1cn(C)nn1)NC(=O)C=CC(C)(C)C 42667,Cc1cnn(CC(N2CCC2CNC(=O)CCC2CCC(C3CC3C)O2)=O)c1 42668,C#Cc1cncc(C(N2CCN(C(=O)C(C)(C=C)CC)CC2CC(=O)NC)=O)c1 42669,N1(C(Cc2nc(CC)sc2)=O)CCCC(C(C)NC(=O)C=Cc2ccsc2)C1 42670,c1(C(N2C(C)CN(C(=O)Cc3cnns3)CC2)=O)cc2c(nc1N)CCC2 42671,c1(-c2n(CCC)nc(CCC(F)(F)F)n2)ccc2c(c1)C(C)(C)CO2 42672,Cc1ccc2oc(C(=O)NCCCN(C(=O)Cc3ccsn3)CCO)c(C)c2c1 42673,C1(NC(c2cn(C)nn2)=O)CCOC12CCN(C(C1CC(F)C1)=O)CC2 42674,C1(NC(Cc2n(C)ncc2)=O)CCC12CCN(C(c1ncc(F)cc1F)=O)CC2 42675,CC(CO)CCCN=c1[nH]c(=NCC2CCN(CC(F)F)C2)c2sccc2[nH]1 42676,C(=O)(CC(C)CCC=C(C)C)NCC1CC(NC(c2cncc(OC)n2)=O)C1 42677,N1(C(c2ncc(OC)cn2)=O)CCC(C2CC2)C1CNC(=O)C=C1CCCC1 42678,N1(C(c2ncccc2O)=O)CC(C2CCCCN(C(=O)C(F)OC(F)(F)F)C2)C1 42679,c1(NC(=O)CC2(O)CN(Cc3cc[nH]n3)C2)ccc(Cl)c(Br)c1 42680,Cc1cccn2c(C(=O)NC34CCCC(NC(C5COC(=O)N5)=O)(C3)C4)cnc12 42681,c1(CCC(=O)NCCOCCNC(=O)CC(F)F)ccccc1OC(F)(F)F 42682,C1(NC(c2c(C)cccc2Cl)=O)COC2C(NC(C3CC(F)(CO)C3)=O)COC12 42683,c1(SC2COCCN2C)ccc(F)cc1.C12CCCN1C(=O)C1(CC1)CN(C)C2 42684,C(=O)(CC(C)CCCCC)N1C(C2CCN(C(COCC=C)=O)CC2)CCCC1 42685,CN1CC2(CC2)CC1C(=O)NCC1CN(C(=O)COC2(C)CCC2)C(C)(C)C1 42686,N1(CC(N2CCC(C(=O)NCCC(=O)OCC)C2)=O)CCCCC1C 42687,C1(NC(c2cn[nH]c2)=O)CC1C1CCN(C(=O)C(=CC2CCCCC2)F)CC1 42688,CCC(CC(=O)N1CC2CCC(C(=O)N(c3csnc3C)C)(C2)C1)C(C)C 42689,C1(C(=O)NCC(C)(C(C)C)NC(Cc2c(C)noc2C)=O)C(O)C(=O)N(C)C1C 42690,c1(C(N2CC(NC(C3C(C)(C(F)(F)F)C3)=O)C2)=O)c(C2CC2)nc2sccn12 42691,N1(C(=O)Cc2ccsc2)CC2=C(C1)CN(C(C1CC1c1ccccc1OC(F)F)=O)C2 42692,Cc1ccc2[nH]cc(C#N)c(=NCc3c(F)cccc3Br)c2c1 42693,Cc1c(F)ccc(C(N2CCC(CNC(C3CN(C4COC4)C3)=O)CC2)=O)c1C 42694,c1(NC(C23CC2CN(C(c2onc4ccccc24)=O)C3)=O)ncnc2sc(Br)cc12 42695,Cc1n[nH]c(C)c1C(C)CC(=O)NCC(F)CNC(=O)CCC(F)F 42696,S(=O)(=O)(CCC1CCc2ccccc21)N1C(C)CC2(CCC2)C1 42697,C(c1ccccc1C)=CC(N1C(C)(CNC(CCSCCC)=O)CCC1)=O 42698,C12(C(=O)NCCC(=O)OCc3ccsc3)CC(CO1)N(c1ncccn1)C2 42699,CC(CN(C)C)CCC(=O)NCC(C1CCC1)NC(=O)CSCCC#N 42700,CC1(C)CN(C(c2ccsc2Cl)=O)CCC1NC(=O)CCCC1CC1 42701,C1(C)(CNC(Cc2c(CC)con2)=O)CCCN(C(c2cc(OC)cs2)=O)C1 42702,CCCCC#CC(C)(C)NC(=O)C(C(C)C)NC(=O)CC1=CCOCC1 42703,c1(CC(=O)NC2CCC(CCNC(CC=C(C)C)=O)C2)ccc2nn[nH]c2c1 42704,C1(C(N2CC3C(C(N4CC(CC)C4)=O)C3C2)=O)CCc2ccccc2C1 42705,N1(C(C(=O)NCC(C2COC(C)(C)O2)O)=O)CCC(=C(Br)Br)CC1 42706,Cc1cccc2[nH]c(-c3ccnc(NC(c4ccccc4[N+](=O)[O-])=O)c3)cc12 42707,C(=O)(C(C)(F)C(F)(F)F)N1CCC(CCN(C(C2(C)CN(C)C(=O)C2)=O)C)CC1 42708,N1(C(C2(CSC)CCC2)=O)CCCC(NC(c2nnc(O)cc2O)=O)CC1 42709,C(c1nc2ccccc2s1)=C(C)COc1ccc(C)c(OC(F)(F)F)c1 42710,CC1(F)CC(C(=O)NC(C(=O)NCc2nn[nH]c2C2CC2)c2ccoc2)C1 42711,N1(C(CS(=O)(=O)N(CC)CC)=O)CC(OC)CC(NC(c2cn[nH]c2)=O)C1 42712,c1(N2CCC(N(C(C3CC(=O)CC(=O)N3)=O)CC)C2)[nH]c(=O)n(C)c(=O)c1C#N 42713,N1(C(C=CCN(C)CC)=O)CCN(C(=O)CN2CC(C)(C)C2)CC1CS(C)(=O)=O 42714,C(=O)(C(C(C)C)C(C)C)NC1C2(CN(C(c3ccc(NC(=O)OC)cc3)=O)C2)C1 42715,C1(COC)CCN(C(c2csc(CNC(c3ccc(Cl)s3)=O)c2)=O)CC1 42716,c1(OC)ccc(C(=O)NC(C)CCNC(C2CCN(C)C2=O)=O)c(F)c1F 42717,C(CC1=CCCCCC1)NC(=O)CC1CCN(C(C2COC(=O)N2)=O)C1 42718,O=S(=O)(c1ccc2[nH]ccc2c1)NC1CCCNCC1F 42719,c1(C(=O)NC(CC=C)CNC(=O)CC(C)C)ccn2cnc(C)c2c1 42720,C(=O)(CCCCCn1cc(-c2cnn(C(C)C)c2)nn1)N(C(C)(C)C)CCC 42721,C(=O)(C1=CCN(C(c2csc(CO)n2)=O)CC1)NC1(CC)CCCC1 42722,N1(CCC)CCCCC1C(=O)NC1CCC1NC(c1ccn(CCN(C)C)n1)=O 42723,C1(C(=O)NC2CC(NC(=O)Cc3ccon3)C2)COc2cc(Cl)ccc2C1 42724,N1(C(C(C=C)(C)CC)=O)CCC2(CCCN2C(C2CC(F)(F)C2)=O)C1 42725,c1(C(=O)NC(CNC(CN(C)CC)=O)CC(C)C)cnc2n1CCS2 42726,c1(CC(=O)NC2CC(C)(NC(C(C(C)(C)C)=O)=O)C2)ccc2ccccc2c1 42727,C1(c2cn(CC3N(C(=O)CCOC4CCC4)CCC3)nn2)CC2CCC1CC2 42728,C12(C(N3CC(CNC(C=C(C)C)=O)C(C(F)(F)F)C3)=O)CCN(CC1)S(=O)(=O)C2 42729,CC(C)(Cc1cnn[nH]1)C(=O)N1CCC(CNC(c2ccc(C(F)F)cc2)=O)C1 42730,n1(CC)cnnc1C(=O)NC1CC1CNC(=O)C(C)OCCOC 42731,c1(C(N2C(CNC(CCC#C)=O)C(C)(C)CC2)=O)ccc2c(c1)OCCC2 42732,N1(C(C(CO)OC)=O)CCC(C(F)F)(CNC(=O)CCc2ccncc2)C1 42733,c1(Nc2cc(N3CCC(C(N)=O)(NC)CC3)ncn2)cccc2c1nnn2C 42734,C(=O)(C1CCc2ccc(OC)cc21)N1CCC(NC(C(CC)C(C)O)=O)C(C)C1 42735,c1(N2CCCC(=O)CC2)nc(NC2CCC3(C2)CC3(F)F)c2ccsc2n1 42736,C1(C(=O)NCCC(C)NC(C2CCC3CC2C3(C)C)=O)CCC2CCCCC2C1 42737,c1(OC)ccc(C(N2CCN(C(=O)C=C(C)c3ccco3)CC2C)=O)c(OC)n1 42738,S(=O)(=O)(CCC(=O)NC1CN(C(c2ccc(CO)cc2F)=O)C1)NC(C)(C)C 42739,C1(OC)CC(NC(c2cc(C)ns2)=O)C12CCN(C(=O)Cc1cnc[nH]1)CC2 42740,C(=O)(C(C)(C)C(C1CC1)NC(C(C)(C)CO)c1cccnc1)OC 42741,C1(C(=O)NC2CN(C(C(=O)NCCOCCCC)=O)C(C)C2)CCCC(=O)N1C 42742,C1(NC(C2CC2C2CCC2)=O)CC2CC1CC2C(N1CCC1C1CCCCC1)=O 42743,CC(C)C(C(=O)NCC(=O)NCC(N1CCOCC1)=O)NC(N)=O 42744,N1(C(=O)CC2CCCOC2)CCC(S(=O)(=O)N2CCCC2)CC1 42745,N1(C(C(C)N(C(C)=O)C)=O)CC(NC(C2CCC2)=O)C2(CCC2)C1 42746,c1(C(=O)NCCN(CCC)C(c2cnc(C(C)C)o2)=O)c(C)coc1C1CC1 42747,c1(CC(=O)NCC(CCC)NC(=O)CSC(F)F)cccc(C)c1 42748,c1(CN(CC(C)C)Cc2ncc(-c3cccc(Cl)c3)o2)ccc(Cl)cc1 42749,N1(C(c2nnn3c2CSCC3)=O)CC2(CCN(C(C3CC(=C4CC4)C3)=O)CC2)C1 42750,C1(CCC)(NC(C2CC(=O)NC(=O)N2)=O)CCCN(C(c2ccnc(C)n2)=O)C1 42751,Cc1nncc(C(=O)NC(CCN(C)C)C(=O)N(CC(O)C2CC2)C)c1C 42752,N1(C(C2ON=C(CC)C2)=O)CCN(C(=O)Cc2ccc3c(c2)CC3)C(C2CC2)C1 42753,C1(NC(COC)=O)COC2(CCN(C(c3ccc4c(C(=O)OC)n[nH]c4c3)=O)C2)C1 42754,c1(CCC(=O)NC(C)CN2CCC(F)(F)C2)ccc(Br)c(Cl)c1 42755,N1(C(COCCCC)=O)CC=CC(C(=O)NC(c2ccncc2)CC)C1 42756,C1(C)(COC)CC(NC(c2c(C)cnn2C)=O)CN1C(c1scnc1Cl)=O 42757,C1(NC(c2c(CC)c[nH]n2)=O)CN(C(=O)Cc2ccco2)CC12CC2 42758,CCCCCCCC(=O)N(C)CC1CN(C(=O)CC2CC(CC)C2)CCO1 42759,Cc1cocc1NC1(C(=O)NCCOC2CN(C(=O)CC)C2)CCSC1 42760,c1(OC)ccc(C=CC(=O)NCCCCCCN(C(=O)CC(C)CF)C)cc1O 42761,N1(S(CC(=O)OCC)(=O)=O)CC2CCCC2(NC(C)(C)C2CC2)C1 42762,C1(CC(=O)NCCC(=C)CNC(=O)Cn2ncc(Br)c2C)CC2CCC1C2 42763,c1(CCC(=O)NC(C)CNC(C23CCCC2C3)=O)ccc2ccccc2n1 42764,C1C(C)CNC(=O)N1C.C(=O)(CCNC(=O)C=CCl)NC1C(C(C)O)C1 42765,C12CCCCC1N2.c1(NC(=O)CSc2cnco2)ncccn1 42766,c1(NC(c2c(COC)n(C)nc2)=O)nccc2[nH]ccc12.C(C(C)(C)CC1CC1)O 42767,c1(NCCCCOC(C)C)cc(=NCC2CS(=O)(=O)CCO2)[nH]cn1 42768,C1(C(N(C2CCCC2)CC=C)=O)CCC(C)(C)N(C(C2CC2(F)Cl)=O)C1 42769,C(=O)(C1C(C)(C)OC(=O)N1)OC.N1(C(C(=O)OC)=O)CCC(c2noc(C)n2)CC1 42770,c1(NC(N(C(CC(=O)OCC)Cc2ccccc2)C)=O)ccc(F)cc1F 42771,CCCC(C)CN=c1cc(NCc2ccccc2CC)nc(COC)[nH]1 42772,c1(C(=O)NC2CN(C(Cc3cccc(OC)c3)=O)C(C)C2)cccc2nn[nH]c12 42773,N1(C(C2(NC(=O)CCC3OCCO3)CCCC2)=O)CCC2C(C1)C2(F)F 42774,c1(C(=O)OC)cc(C(=O)NCC(C)NC(c2cscc2F)=O)n2c1COCC2 42775,c1(C(N2C(CNC(C(C)Oc3ccccn3)=O)CC2)=O)cccc(C(N)=O)n1 42776,c1(C(CC)(C)O)cn(CC2CN(C(c3coc(CS(C)(=O)=O)n3)=O)C2)nn1 42777,CC1(C)CC(O)CN1C(=O)CN(C1CCCC1)C1CCCC1 42778,CCC(C)(C)C(O)C(=O)N1CCCCC(C(=O)NC2CN(C(=O)C3CC3)C2)C1 42779,c1(N2CCC(CCNC(C(C(C)C)(C)O)=O)CC2)ncc([N+](=O)[O-])cc1C(N)=O 42780,c1(C(=O)NC(C)C(C)NC(=O)C(C)(C)CS(N)(=O)=O)cc2c(cc1Cl)NC(=O)C2 42781,c1(CC)cc(=NC(=O)C2CCN(C(=O)C(CC3CC3)OC)C23CCC3)[nH]n1C 42782,c1(NC(C)=O)ccc(C(N2CCCCC2C(N2CC3CC3C2)=O)=O)cc1 42783,Cc1n[nH]c(C)c1CC(N1CC2C(CN(C(=O)C(C)(C)C)C)C2C1)=O 42784,C1(CNC(C(C)NC(C)=O)=O)CC(F)(F)CN1C(=O)COC1COC1 42785,Cn1ncc2c(N3CC4CC4C3)[nH]c(=NCCCN3C(=O)CNC3=O)nc12 42786,CC1CCC(CNC(C2CCCCC2)=O)CN1C(=O)COC1(C)CCCC1 42787,c1(C(=O)NC(CNC(C(C)(C)OCC)=O)C)cccc(C)n1 42788,c1(SCC)ncc(Cl)cc1C(=O)OCC(C(C)C)OCC1CC1 42789,C1(NC(C(CC)OCC)=O)CCN(C(=O)Cn2nnc(C3CC3)n2)CC(C)(C)C1 42790,C12(NC(C(CC#C)CC#C)=O)CCCC1(F)CN(C(=O)C(C)COCC)C2 42791,Cc1nnc2c(C(=O)NC(C)C(C)NC(c3ccncc3N)=O)cccn12 42792,c1(C(c2nnnn2C2CC2)NCC=CCSC)cccc(C(F)(F)F)c1 42793,n1(NC(=O)CCCn2cc(C)cn2)cc(C)nn1.C12(CC1)CC(=O)NC2C.CSC 42794,C1(CN(C)C)COCCN1C(=O)CC(C1CC1)NC(=O)C(C)(C)C1CCOC1 42795,C(=O)(C1=CC2CC(C1)CC2O)NC(CN(C(Cn1nc(C)oc1=O)=O)C)C 42796,S(=O)(=O)(c1ccc(F)cc1Cl)NCC(N1CCOCC2(COC2)C1)=O 42797,C1(C2CC2)(CNC(=O)CC2CC=CC2)CCN(C(=O)CN2CCCCCC2)C1 42798,c1(OCC)ccc(C(C)NC(=O)CCC2(C)CC2)cc1F 42799,CC(CC(F)(F)F)C(=O)NC1CCN(C(=O)C=C2CCSCC2)CC1O 42800,c1(C(N2CCCCC2C#N)C(=O)NCCCC)cnc(Br)c(Cl)c1 42801,CCCC(C)(CCC)C(=O)N1CCC(CNC(=O)CN(C)C)(OC)C1 42802,c1(NCC#CC)cc(=NCC(C(C)C)c2ccnn2C)[nH]cn1 42803,C1(C(=O)NC(C2(C(N(CC)Cc3cccnc3)=O)CC2)C)CCN(C)CC1 42804,c1(C(=O)NC2CCN(C(CC(C)C3CC3)=O)C2(C)C)ccc2[nH]ccc2c1 42805,CCC(CC1CC1)C(=O)N1CC(NC(=O)CCN(C)CCO)C(F)C1 42806,Cc1nc(CCCC(=O)NC2CC(NC(c3cscc3C(F)F)=O)C2)cs1 42807,C1(CC)C(C(NC[Si](C)(C)C)=O)CCCN1C(c1ccccc1F)=O 42808,N1(C(c2cnns2)=O)CCC2(CCCN2C(c2cc(Cl)n[nH]2)=O)CC1 42809,C1(CNC(C(=O)NCc2ccc(-n3c(C)cc(C)n3)cc2)=O)CC2CCCC2C1 42810,N1(C(c2n(C)cnc2)=O)CCc2sc(CNC(=O)CCc3cnc(O)[nH]3)nc2C1 42811,c1(C(N2CCC(COC)(NC(=O)CC(O)CN(C)C)C2)=O)cc2occc2n1C 42812,C1(CN(C(C2CC(C)C2)=O)C)CCCC1NC(=O)C(CN(C)C)c1ccccc1 42813,CC1CN(C(C2(NC(c3nnn(C(C)(C)C)n3)=O)CC2)=O)CC(CCC2CC2)O1 42814,C1(CC)CC(C)CN(C(=O)CC(C)(C)NC(=O)CCCN=[N+]=[N-])C1 42815,c1(C(=O)NC(CC(=O)N(C23CC(C2)C3)CC)C)cnn2c1OCC2 42816,C1(c2nnnn2C)(Nc2ncc(-c3ccc(Cl)cc3)o2)CSCCSC1 42817,N1(C(CSS(C)(=O)=O)=O)CC(NC(=O)Cc2cc(-c3ccccc3)on2)C(F)C1 42818,c1(C(=O)NC2CC2NC(c2ccc(OC3CC3(F)F)cc2)=O)ccc[n+]([O-])c1 42819,C1(C(N)=O)CN(C(=O)C(=O)NCc2cc(N3CCCC3)n[nH]2)c2ccccc2O1 42820,c1(C(N(CCCN(C(CCNC(C2C(C)C2)=O)=O)C)C)=O)scc2c1CCCC2 42821,C(=O)(CC(C(C)C)C(C)C)NC(CCNC(C1CN(CC)C(=O)C1)=O)(CC)CC 42822,Cc1cnn(C)c1CC(N1CC(N(C)C(C2C3COCC23)=O)C1)=O 42823,C1(CC)C(NC(=O)CNC(=O)CC(C)(C)C)CCN1C(=O)CC1CC(C)C1 42824,C1(CNC(CNC(CC(C)C)=O)=O)CC(C)(C)CN1C(c1cc[n+]([O-])cc1)=O 42825,c1(OC)c[nH]c(C(N2CC(NC(=O)C(C)NC=O)C(O)C2)=O)cc1=O 42826,CCC(C)C(O)C(C)C(=O)N1CC(NC(=O)CCCCCC(C)C)C(O)C1 42827,N1(C(c2n(COC)ncc2)=O)CC(NC(=O)C=CCCC(C)C)CC(C)C1 42828,CC12CC1CN(C(=O)C(N1CCN(c3cccc(Br)c3)CC1)=O)C2 42829,c1(C(=O)NC2CC(CNC(C(CC)O)=O)C2)ccc(C(C)C)cc1 42830,N1(C(C(CC)OCC)=O)CCC(CC(=O)NCC(C)(C)CC)C1(C)C 42831,C1(C)(C(N2C(COC)CCCC2)=O)CCCN(Cc2ncccc2C)C1 42832,O=C(CCCc1ccsc1)NCC1CC(Sc2ccccc2)C1.c12nccn1C2 42833,C=C=CCCC(=O)NCCCOCC(c1ccccc1)NC(=O)CCC1CC1(C)C 42834,C(C(C(=O)N(C)CCN(C)C1CC1)C(C)C)NC(c1c(C)n(C)cn1)=O 42835,c1(CCC(=O)NCCC(CNC(=O)Cc2cnoc2)O)nnc(S)nc1O 42836,S(=O)(=O)(c1ccnn1C1CCC1)N1CCN(C(=O)Nc2ccsc2)CC1 42837,C(C(O)CS(C)(=O)=O)NC(N(C(c1onc(C)n1)C)C)=O 42838,C(=O)(CC(C)(C)CCC)NCC(CC=C)C(=O)NC1COCC1O 42839,C(=O)(CCCC(C)=O)N1CC(NC(C(C)=CC)=O)C(c2nccn2C)C1 42840,C1(C(=O)NCCN(CCC)C(c2cc(O)nn2C)=O)OCCOC12CCC2 42841,N1(C(=O)OC(C)(C)C)CCC(C(C)(O)CNC(c2cc(CC3CC3)ns2)=O)CC1 42842,C1(C(=O)NC(CC)CNC(C2CC(F)(CC)C2)=O)COCCN1CC 42843,C=CC(C)CC(=O)NC1CC(C(=O)NCc2ccccc2CC)CC1O 42844,O=C(C1=CCN(C(=O)COC(F)(F)F)CC1)NC1CC1C1CCCC1 42845,C(=O)(C(F)(F)C1=CCOCC1)N(C)CC1CCN(C(=O)C(F)(F)C(O)C2CC2)C1 42846,c1(CCC)sc(C(=O)NC2CC(CNC(C3CCN(C(=O)OC)CC3)=O)C2)cc1C 42847,C1(C(=O)NC2C(C)CCN(C(C=C(C)C)=O)C2C)CCc2nc(O)[nH]c2C1 42848,c1(CC(=O)NCC(CNC(=O)CC2CCCCC2O)OC)ncc(F)cc1F 42849,C1(C(N2CCC(CNc3cc(Cl)ncn3)C2)=O)CCCCC1n1cccn1 42850,C(=O)(C(F)(F)C(F)(F)OC(F)(F)F)N1CCN(C(C)=O)C(c2nccn2C)C1 42851,C1(CC(N2CCC(C(=O)NCC)C2)=O)CCN(S(=O)(=O)Cc2ccccc2)C1 42852,c1(C(=O)NC2C3CN(c4c(C#N)nccn4)CC32)cc2cc(Cl)cnc2[nH]1 42853,C(CCCC(=O)NCC1CCCCN1C(c1cccc(F)c1SC)=O)(OC)OC 42854,N1(C(C(CCSC)OC)=O)CC2CC3CC2C1C3NC(=O)C(c1ccc(Cl)s1)C 42855,c1(CN2CC(NC(c3c(O)cccc3F)=O)(CO)C2)c(O)ccc(Cl)c1Cl 42856,N1(C(CSCC#C)=O)CCN(C(=O)Cc2ccc(F)cc2)C(c2nccn2C)C1 42857,c1(-c2ccc(-c3n(CC(CC)CO)ccn3)s2)cc(-c2ccccc2)n(CC)n1 42858,Cc1cc(C(N2CC3CC3(CNC(=O)OC(C)(C)C)C2)=O)cnc1C 42859,Cc1ccc(C(=O)NCC2COC(CNC(=O)Cc3csc(Cl)c3)C2)cc1CO 42860,C(C(C(=O)N1CCC(C)(NC(c2cccnc2)=O)C1)C(C)(C)C)OCC=C 42861,c1(C(=O)NC(CC)CN(C(=O)C(CO)NC(N)=O)C)ccc2c(c1)NC(=O)CC2 42862,C1(C)(CC(=O)N(C)CC2(O)CN(C(CC3CCCN(C)C3)=O)C2)CCS(=O)(=O)N1 42863,C(=O)(C(C)(C)C(=O)NC(C1CC1)C1CC1)N1C(C)CC1C(=O)N(C)C(C)(C)C 42864,Cn1ncc2cc(C(N3CC(NC(C4C=CCC4)=O)CC(F)C3)=O)sc12 42865,CC(C1CC1)=C(F)C(=O)NC(C)C(C)NC(C1(CN(C)C)CC1)=O 42866,c1(OC)ccc(C(N2CC(CNC(c3cc(C#N)c[nH]3)=O)C3CC23)=O)cc1Cl 42867,CCS(=O)(=O)c1ccc(S(=O)(=O)NC2C(C(=O)O)C3CCCCCC23)cc1 42868,C1(CCNC(C(n2ncc(C)c2)C)=O)CCCN(C(c2ccc(F)nc2)=O)C1 42869,C(CC(=O)NC(C)CNC(=O)CCC1CC1(Cl)Cl)N(C)C(=O)OC(C)(C)C 42870,c1(CS(N2CCC(Oc3ccc(C)cc3)CC2)(=O)=O)nc2ccccc2[nH]1 42871,N1(CC)CCC(NC(=O)CCN(CCO)C(C2(C(C)(C)C)CCC2)=O)CC1 42872,N1(C(c2cc(OCC)ncc2)=O)CCCC(NC(c2ccncc2)=O)C(F)C1 42873,C1(C(N2C(CCC)CN(C(=O)CC(C)(C)C)CC2)=O)Cc2cncn2C(=O)N1 42874,C#Cc1c[nH]nc1C(=O)NC1CN(C(c2csnc2C2CC2)=O)CC1O 42875,c1(C(=O)NCC2C(NC(c3ccc(CN(C)C)nc3)=O)CC2)cc2ccsc2s1 42876,N1(C(C2CCC(C)(O)CC2)=O)CC2CC(C(=O)NCCCCC(F)(F)F)C(C2)C1 42877,C1(NC(CC(=O)N2CC(N(C(C(C(C)C)F)=O)C)C2)=O)CC(C)CC(C)(C)C1 42878,C(=O)(CC(=O)NC1COCC1NC(=O)C(O)Cc1ccccn1)N(CC)CC 42879,C(=O)(C(CCCOC)NC(=O)Cc1cnns1)NC(C#C)(CC)CC 42880,c1(C(N(C2CCN(C(=O)CCc3nncs3)C2)C)=O)ccnc2ccc(O)cc12 42881,C1(C(=O)NC)CCN(C(C2(CCNC(c3cc(C)[nH]n3)=O)CCC2)=O)C1C 42882,C1(C(=O)NC)CC(F)(F)CN1C(c1cc(-n2cc(C(C)(C)O)nn2)ccc1Cl)=O 42883,c1(CC(=O)N(CC(C)NC(C(CC#C)(C)CC)=O)C)ccc2ccccc2c1 42884,c1(OC)cc(C(=O)NC2CC2NC(C2CC(C)(O)C2)=O)ccc1O 42885,C#CCCC(C(=O)NC1CCCC(O)C1O)NC(C1COCC(C)O1)=O 42886,C(C(=O)N1CC(NC(=O)C(C)(C)C#N)C(c2ccnn2C)C1)(C(C)C)SCC 42887,CCC(C(=O)N1CC(NC(C2(n3cccc3)CCCC2)=O)C1)NC(N)=O 42888,C=CC(C)(CC)C(=O)NCC1CCN1CCc1ccc(-n2cccn2)c(C)c1 42889,c1(C(=O)NC(C2N(C(C(COC)OC)=O)CCC2)C)n[nH]c2ccc(OC)nc12 42890,C1(CC=C)(NC(c2ccnn2C)=O)CN(C(c2cc(C(C)(C)C)c[nH]2)=O)C1 42891,N1(C(C=C2CCC(C)CC2)=O)CC2=C(C1)CN(C(C1CC1(C)C(F)F)=O)C2 42892,c1(C(=O)NCC2(O)CC(NC(CCS(C)=O)=O)C2)c(F)cccc1Cl 42893,c1(SC)ccc(N)cc1C(=O)NC(C)C(C)NC(=O)Cc1csc(C2CC2)n1 42894,C(=O)(C(C)C(O)C(C)CC)N1CCC(C(=O)NCC(C#C)OC)C12CC2 42895,n1(CC(=O)NCC2CC(F)(CNC(C3CC(=C)C3)=O)C2)cc(C#N)cn1 42896,C1(O)(CNC(C(C=CC)O)=O)CCN(C(=O)Cc2ccccc2C)C1 42897,N1(C(C2CCC(C)(CC)O2)=O)CC2CCCC(C1)N2C(c1cc(C(F)F)cs1)=O 42898,c1(C=O)ccn(CCNC(=O)CN(C)C2CC2)c1.C(C)(CNC)SC 42899,N1(C(C(C)NC(=O)NC)=O)CC(CNC(=O)CCn2cc(Cl)cn2)C(C)C1 42900,N1(C(Cn2cc(COC)nn2)=O)CCN(C(c2cncnc2C)=O)CC(O)C1 42901,CC(C)S(=O)(=O)CC(=O)N(CCCNC(=O)CP(C)(C)=O)C 42902,N1(C(c2c(C)nsc2)=O)CCN(C(C2CC(C(F)(F)F)C2)=O)CC(CO)C1 42903,CC(c1ccccc1OC(F)F)=CC(=O)NCC1CC1CNC(C1CCOC1)=O 42904,N1(C(CC2C(C)(C)OCCO2)=O)CCC2CN(C(=O)C=CC=C(Cl)Cl)CC2C1 42905,Cc1cc(C(=O)NCC(CC(C)C)NC(C2CCC(F)CC2)=O)cnn1 42906,c1(NC)ccc(C(=O)NCC2(C(=O)NC(C3CCCO3)CO)CCCCC2)nc1 42907,c1(CNC(=O)NC(CCC)CCC)nn(C)c(C)c1Cl 42908,N(C(=NCCC(C)C)NCC1(C)CCC(NC(C)=O)CC1)C1CN(C(=O)OC)C1 42909,C1(C(=O)NCC(CC(C)C)NC(C2C=CCS2)=O)CC(C2CCCC2)C1 42910,C1(C)(C(=O)NC2CC(CNC(C(C)Sc3nncn3C)=O)C2)CC(F)(F)C1 42911,C1(C(N2CCOCC2)=O)CCCCC1NC(CN(C(=O)C(O)C1CCCC1)CC)=O 42912,C1(CC(=O)NCC2C(C)(C)CCCN2)CCc2ccccc2N1 42913,N1(C(c2scc(C)n2)=O)CCC(O)C(C(N2CCC(c3ccncc3)C2)=O)C1 42914,N1(C(C(COC)OC)=O)CCC(C)C(NC(c2cc(-c3cn(C)nn3)on2)=O)C1 42915,c1(C(C)NC(C23CC(NC(c4c(CC)c[nH]n4)=O)(C2)C3)=O)ccc(Cl)cc1 42916,CCCCCCC(CC)(CC)C(=O)NCC(CNC(=O)CCCOC)C(F)(F)F 42917,C1(CCNC(=O)NC2CC(CC(=O)OC)C2(C)C)CCC(F)(F)CC1 42918,C(C)(C(C)S(C)(=O)=O)N(C(C(=O)NC1CN(C(C)C)C(=O)C1)=O)C 42919,N1(CCCOC)CCCC1C(C)(C)CNC(c1cnc(N(C)C)o1)=O 42920,c1(CNC(Cc2c(C)nn(C)c2)=O)n[nH]c2c1CN(C(=O)C(C)S(N)(=O)=O)CC2 42921,c1(C(N2CCCC(NC(C34CC5CC3C4C5)=O)C2)=O)ccc2ncccc2c1 42922,C1(O)(C(=O)NCC2(CC)CN(C(=O)CCCC(C)(C)C)C2)CCCC(C)CC1 42923,c1(CCC(=O)NC2(C)CC(NC(=O)Cc3cnoc3)C2)cncc(F)c1 42924,c1(C(=O)NC2CC(F)(CNC(C3(C)CCN(C)C3)=O)C2)cccc2nc(O)[nH]c12 42925,c1(CC)cc(C)[nH]c(=NCC2CC3(CC(NC(=O)Cc4csc(CC)n4)C3)C2)n1 42926,N1(C(c2ccc(SC)nc2)=O)CCCC(O)(CNC(c2cc(C3CC3)on2)=O)C1 42927,c1(C(=O)NC(C(=O)NCCc2ccc(C)s2)C2CC2)cnc(C)c(C)c1 42928,c1(C(=O)NC(CN(C(c2cccc3ncnn23)=O)CC)C)ccc(O)c(F)c1F 42929,c1(C(N(C(C)C)CCNC(=O)C(F)F)=O)ccc(N2CCCCCC2)nc1 42930,N1(C(C2CCCCC2)=O)Cc2ccnn2CC(NC(C2CC23CCC3)=O)C1 42931,C(C(C)C(=O)NC1COCC1NC(c1cc(C(N)=O)c[nH]1)=O)OCC 42932,C1(C(C(=O)NCCCN(C)C(C2(C)CCCN2C)=O)(C)C)CCC(O)CC1 42933,c1(C(CC)C(=O)N(CC(O)CN(C)C(C2(OC)CC2)=O)C)ccc(F)cc1 42934,C12(CNC(c3cc(CC)on3)=O)CCCC1N(C(=O)C(CCOC)OC)CCC2 42935,Cc1cc(C(=O)NC(C)CCNC(=O)Cc2ccncc2Cl)c(Cl)cc1Cl 42936,c1(C(C)=O)cccnc1NC(C1CCC(NC(c2ccccn2)=O)C1)=O 42937,c1(C(N2CC(C(C)CO)C2)=O)ccc2c(c1)CCCN2C 42938,c1(C(=O)NCCN(C(C)C)C(C2CCCCCCC2)=O)ccc2nc(Cl)nn2c1 42939,N1(C(c2ccn(CC#N)n2)=O)CC2=C(C1)CN(C(=O)CCn1cncn1)C2 42940,Nc1c(CNC(=O)NC2CCCC2c2cccc(Br)c2)cccc1F 42941,c1(NC(N2CCCC(C)(C(F)F)C2)=O)ccc2c(N)nccc2c1 42942,c1(C(=O)NCCCC(C)NC(COCCC)=O)cc(Cl)c(F)cc1F 42943,c1(NC(=O)CCO)ccc(C)cc1.N1(C(CCNS(C)(=O)=O)=O)CC(C)(CCOC)C1 42944,C1(NC(C2CC(C3CC3)C2)=O)CCOC(C(N2CC(O)(c3cc[nH]n3)C2)=O)C1 42945,C(C(=O)NCC12CCC(CC1)N2C(C1CCCOCC1)=O)(C(C)(C)C)SC 42946,c1(CCCC)nc(CN(C2CCCCC2n2cc(COC)nn2)C)c(Cl)[nH]1 42947,c1(SC)cc(C(=O)NCC2C(C)CCCN2C(=O)CC(=O)NC2CC2)ccc1F 42948,CC(C)(CNC(=O)COCC(=O)NC(=O)Cc1sccc1Br)CC1CC1 42949,CCC(C(=O)N1CC2C(NC(=O)Cc3scnc3-c3cccs3)C2C1)C(C)(F)F 42950,C(CCC(F)(F)F)N(C(CC1N(C(Cc2c(C)con2)=O)CC1)=O)C 42951,c1(C(N(CCCCCC)CCNC(=O)C(C)C#N)=O)ccc2nonc2c1 42952,CC(C)CC(C)(CNC(=O)C(C)(C)c1ccno1)NC(c1cc(C(C)C)on1)=O 42953,c1(C(N2C(CNC(CCC=C(C)C)=O)C=CC2)=O)cnc2ccnn2c1C 42954,Cc1ccc2oc(C(=O)NC(C)(C)CCCNC(C3(CO)CCC3)=O)cc2c1 42955,CC(C(=O)NCCSCC(=O)NCC(=O)NC(C)C)=CC1CC1 42956,c1(CC(=O)NC23CC(C(=O)NCC4CCCSC4)(C2)C3)ccccc1F 42957,C1(N(C(C(CNC(c2nc(C(C)C)oc2)=O)O)=O)C)CCCC1(C)O 42958,Cc1cc(Cl)cc(C(=O)NCCCNC(c2n[nH]c3c2CSCC3)=O)c1C 42959,CCC(CC)CCCNC(=O)CCC1CC1COC 42960,c1(C(=O)NC2C(CNC(=O)CCC3OCCO3)CCC2)cccnc1C(F)F 42961,N1(C(C2C(C)(Br)C2)=O)CCCC(C2CC2NC(c2cnn(CC3CC3)c2)=O)C1 42962,c1(C(=O)NCC2C(NC(C=CC(C)C)=O)C2)cccc(C2CC2)n1 42963,Cn1nc2c(c1CNC(=O)CCCOc1ccc(I)cc1F)CCCC2 42964,C(=O)(C(C)CC(F)(F)F)NC(c1occ(C(N(CC(C)C#N)CC)=O)n1)C 42965,C(=O)(CCn1ccnc1)N(CC(C)O)CCNC(=O)CC1(C(F)(F)F)CC1 42966,c1(SC(C)C(N)=O)ccc(C(=O)NC2(C)CN(C(c3ccncc3)=O)C2)cc1 42967,c1(-c2n(-c3c(C)cccc3C)nc(C(C)C3CC3)n2)sc2cccc(F)c2c1C 42968,c1(C(N2CC(NC(=O)C(F)(F)CC3CC3)CC(C)C2)=O)nc2cccnc2s1 42969,CCCCC(CNC(C1CCCN1C)=O)NC(c1snc(Cl)c1Cl)=O 42970,N1(C(=O)Cn2cc(CC3(O)CCC3)nn2)CCC(n2ccc(C(=O)O)n2)CC1 42971,c1(CNC(CC(C)SC)=O)ccc(C(=O)NC2CCOCC2C)nc1 42972,N1(C(CC2C(CC)C2)=O)CCCC(CNC(=O)CCn2cccn2)CC1 42973,C(=O)(CC(COC)COC)NC(CC=C)CNC(C1CCNC(=O)C1)=O 42974,N1(C(CCOC)=O)CC2CCN(C(=O)C#CC3(C)CC3)CC12 42975,c1(OCC(N)=O)ccc(C(=O)NCC(C)NC(=O)C=CSc2ccccc2)cc1 42976,c1(C(=O)NC2(C(=O)NCc3ncccc3F)CC(CO)C2)ccc(O)cn1 42977,C1(NC(c2c(CC)c[nH]n2)=O)CCN(C(=O)CSc2cccc(F)c2)CC1(C)C 42978,C(=O)(C1COc2ccccc21)N1CC(C)(C)OC(CNC(C2CC=CCC2)=O)C1 42979,c1(-c2cn(CCC(=O)N(C3CCC(=O)NC3)CC)nn2)nc(C)cc(C)n1 42980,N1(C(C2N(Cc3c(N(C)C)cccc3)C(C)CC2)=O)Cc2ccc(Cl)cc2C1 42981,Cn1cc(C(=O)NC2CC2CNC(c2ccc(-n3cncn3)cn2)=O)n(C)c1=O 42982,N1(C(c2cncc(SCC)n2)=O)CCN(C(=O)CC=C(C)C)C(C)C1C 42983,c1(C(=O)NCC(CNC(C(CCCC)C)=O)F)ccc(S(N)(=O)=O)cc1Cl 42984,c1(C(=O)NC(C2(O)CN(C(C(CC#C)C)=O)C2)C)cncc(C)c1Cl 42985,N1(C(C(CNC(C=CC(=O)NC(C)C)=O)N(C)C)=O)CCCC(N(C)C)CC1 42986,c1(C(=O)OC)nc(Br)cnc1NC(C1CCC(C)N1Cc1ncc(Cl)cc1C)=O 42987,Cc1c(NC(=O)Cc2ccccc2NCc2ccsc2)ccnc1Cl 42988,C1(C)(C(=O)NCCC(C)CCNC(=O)CCCc2ccccn2)CC2CCC1C2 42989,C1(C(N2C(CNC(c3c(C)scn3)=O)CCCC2)=O)COC2COCC12 42990,c1(C(N2CCC(C)(NC(c3nc(C)c(C)[nH]3)=O)C2)=O)ccc2[nH]c(=N)[nH]c2c1 42991,CCCN=C(NCC(=O)NC(C)CC)NC(c1cc(C)sc1C)C 42992,c1(CC)cc(C(=O)NCC2CC(CNC(=O)C(N)=O)CO2)on1 42993,C(=O)(C(C#N)C(C)(C)C)N1C(C(NOCC)=O)C2CCC1C2.C1(=O)CCCN1 42994,C(=O)(C1=CS(=O)(=O)CCC1)NCC1C(C)CN(C(=O)CCC2CC(F)(F)C2)CC1 42995,N1(C(c2cc(C)sc2)=O)CC(NC(C2(Cc3cnn[nH]3)CCC2)=O)C(C)C1 42996,c1(C(N2CCC(O)CC2)=O)ccc(Br)cc1OC(F)(F)F.c12sccc1NC2=O 42997,C(C)(C(=O)NC1CC(NC(=O)CCc2nc[nH]n2)C1)=CC 42998,N1(C(C2C(C)(Br)C2)=O)C(CNC(=O)Cn2cnnn2)CC2COCC12 42999,C1(NC(CC2(COC)CCCC2)=O)CCC(C)(C)CC1CNC(=O)C=CBr 43000,c1(OC)cc(C=CC(=O)NCCc2ccc(CNC(c3cnn[nH]3)=O)cc2)sn1 43001,Cc1ccncc1C(=O)NCCC1CCC(NC(c2c(C)coc2C2CC2)=O)C1 43002,c1(C(N2CC3CCN(C(c4c(SC)ccs4)=O)C3C2)=O)ccc(C)cc1[N+](=O)[O-] 43003,C(C(=O)NCC(C)(CO)NC(C1CN(C2CCC2)C1)=O)(C(C)C)OC(C)C 43004,N1(C(C(CC=C)C)=O)CCCCC(NC(c2cc(-c3ccc(F)cc3)cs2)=O)C1 43005,c1(C(N(C2CCN(C(=O)CC3CC3(C)C)C2)CC)=O)ccc(C)c2c1NCCC2 43006,c1(C(CN2CC(CC(=O)OC)(N(C)C)C2)O)cccc(OC)c1 43007,c1(C(N2C(CNC(C(CC#C)O)=O)CC(F)C2)=O)cnn2c1NCCC2 43008,c1(C(N(CCCNC(C2(NC(=O)NCC)CCCC2)=O)C)=O)cc(C)ncc1C 43009,c1(CNC(=O)NCC2CCN(C(=O)OC)CC2)ccc2cccnc2c1 43010,CC1CC(CNC(c2cccnc2)=O)CN1C(=O)CCCC1CCCC1 43011,CC1Cn2nc(C(=O)N(c3ccc(OC(C)(C)C)cc3)C)cc2CN1 43012,C#CC1CN(C(=O)C(C(C)OC)NC(=O)C(O)CN2CCCC2)CCO1 43013,N1(C(C(C)CO)=O)CC(NC(c2cncc(F)c2)=O)CC12CCCC2 43014,C1(NC(c2ccc(C)nc2)=O)CC2(CCC(NC(C3C(C)CC3C)=O)CC2)C1 43015,N1(C(CC(C)OC)=O)CCCC(C)(NC(=O)Cc2ccc(O)cc2C(F)(F)F)C1 43016,N1(C(=O)C(O)CCCNC(C23CC2CNC3=O)=O)CCc2occc2C1 43017,Cc1ccc(O)c(CNC(=O)CC=CCNC(c2cn(C)cn2)=O)n1 43018,Cc1ccc([N+](=O)[O-])cc1C(=O)NCC(CO)NC(=O)CCCC1CCOCC1 43019,N1(C(CC2CN(C(C(C)NC(C)=O)=O)C(C)(C)C2)=O)CC2(C1)CC(C)(C)C2 43020,CC1(C(=O)NCCCCNC(=O)Cc2ccc(O)cc2Cl)CCC12CCC2 43021,Cc1ccc(CC(=O)NC2CC(CNC(=O)C(C)CN(C)C)C(O)C2)c(Cl)n1 43022,C=CCC(CC=C)C(=O)N1CC(O)CC1(C)C(=O)NCCCCC 43023,Cc1cnc(CNC(=O)C(c2cccnc2)NC(=O)CN2CCC(C)C2)cn1 43024,c1(OCC)nc(C)ccc1C(=O)NCC(O)CNC(=O)CCc1ccnc(C)n1 43025,c1(C(=O)NC(CNC(C(C)=C2CC2)=O)(C)C2CCC2)ncccc1Br 43026,C1(CC(=O)NC2C(C)N(C(=O)Cc3ccc(CO)cc3)CC2)CCCC(F)(F)C1 43027,c1(C(CC(=O)NCC2CCCN(C(c3cccnc3S)=O)C2)O)ccc(F)cc1 43028,C=CC1(C(N2CCC(C(=O)NC(C#C)CC(C)C)C2)=O)CCCCC1 43029,CCCCC(O)C(=O)N1CC(NC(=O)CCCC(=O)C2CC2)C(C)C1 43030,C1(OC)CC(NC(=O)C(C)CC=Cc2ccccc2)CN(C(=O)CP(C)(C)=O)C1 43031,C1(C(C)C)CN(C(=O)C(O)C(F)(F)F)CCN1C(=O)C(F)=CCc1ccccc1 43032,c1(C(C)C)cnc(O)c(C(=O)NC2CCN(C(C3CC(C)(C)CO3)=O)C2)c1 43033,C1(C(N)=O)CC(F)CN(C(=O)CC2CCN(C(=O)Cc3ccc(O)cn3)C2)C1 43034,N1(C(C(CCC)N(C)C)=O)CCCC2(NC(c3ccoc3Cl)=O)CC2C1 43035,c1(NC(CCC2(C)CN(C(N3CC4CC4C3)=O)C2)=O)cccc(N2CCCC2)c1 43036,C(C(=O)N=S(C)(=O)N(C)C)n1cc(C(C)NC(C(CC)OC)=O)nn1 43037,c1(OC)cc(N2CCCC2)ccc1C(=O)O.S1(=O)(=O)CCNC(=O)C=CC(=O)N1 43038,C1(C(C)C(=O)NCCNS(N)(=O)=O)CCN(C(C2CCN(C)CC2)=O)CC1 43039,N1(C(CCCCSC)=O)CC(C)C(C)(CNC(=O)C(C2CC(F)(F)C2)OC)C1 43040,C#CC1CC2(CC2)CN1C(=O)CCC(C)NC(C1(C#N)CC1)=O 43041,c1(OC)ccc(CC(N)C(=O)NCCO)c(OC)c1.c12cccc(c1)OC2 43042,N1(C(C2(N=[N+]=[N-])CCN(C(c3cc(CC)sn3)=O)C2)=O)CC(C#N)C2(CCC2)C1 43043,N1(C(C(CC)(C)CO)=O)CCCN(C(=O)Cn2cc([N+](=O)[O-])c(C)n2)C(CO)C1 43044,c1(OC)ccc(F)c(CC(=O)NCCC(C)(C)NC(C2CC23CCC3)=O)c1 43045,C1(C(=O)NC(C=CC(=O)NC(C(C)F)C)C)OCC2CCCC12 43046,C1(c2noc(CC(=O)NC(C)CO)n2)(NC(C)=O)CCC(C)CC1 43047,N1(C(C(C)(C)OC)=O)C2CCC1C(CNC(c1nccnc1C(N)=O)=O)C2 43048,CC1=C(C(=O)NC2CCCC2C(=O)Nc2ccc(Br)nc2)CCO1 43049,c1(CNc2c(C)nc(-c3c(OC)cccc3)s2)c(C)nn(C)c1C 43050,c1(NC(C2N(Cc3ccc(SC)s3)CC(F)C2)=O)nc(Br)c(Br)cc1Br 43051,C1(NC(C(CCC)N(C)C)=O)CN(C(=O)CNC(C)=O)Cc2nccn2C1 43052,C(=O)(CC(C=C)CC)NCC(C(=O)N(CC#C)CC#C)CC1CC1 43053,N1(C(c2sc(Cl)cc2Cl)=O)CC(NC(C2(CCF)CC2)=O)CC12CCC2 43054,C1(OC)CC2CC(C(=O)NCCCC(CO)NC(C3(F)CC3)=O)CC12 43055,C1(NC(=O)CCC=CBr)C2CCC1N(C(c1ccc(CF)cc1)=O)C2 43056,c1(C(N(C)CC2CCN(C(c3ccc(F)cc3N)=O)C2)=O)cnc2[nH]ccc2n1 43057,C1(CC(N2CC(O)(CCNC(C(COC)OC)=O)C2)=O)COCC2(CCC2)O1 43058,CCCCC(O)C(=O)NCCC(C)NC(=O)CC(F)(F)c1ccccc1 43059,N1(C(C=C(COC)C)=O)CC(O)(C(C)NC(C2(c3ccccc3)CC(C)C2)=O)C1 43060,c1(CNC(c2n(CC=C)nnn2)c2ncc(Cl)s2)cc(Br)cc(Cl)c1F 43061,C(=O)(C1=CCCCCC1)N1CCC(C)(NC(c2nc(C)n(C(F)F)c2)=O)C1 43062,N1(C(C(C)=O)=O)CCOCC(NC(C2(C(F)F)CCCO2)=O)C1 43063,C1(NC(c2cc(Cl)ccn2)=O)COC2(C1)CN(C(=O)CC1CCC(C3CC3)O1)C2 43064,c1(C(=O)NCC2CC(NC(C(C)C3CCCO3)=O)C2)cc(F)c(N)c(F)c1 43065,N(C1CS(=O)(=O)Cc2ccccc21)C(NC1CCc2c(Cl)cc(Cl)cc21)=O 43066,C1(NC(CSCC=C)=O)CC2CC(NC(C3CCC4CC34)=O)C1C2 43067,C1(NC(CCC)=O)CCCCC1NC(C12CC(CC(C)C)(C1)C2)=O 43068,C1(NC(C(O)N(C)C(=O)OC(C)(C)C)=O)CC2(CCN(Cc3ccno3)CC2)C1 43069,C(C)(CN=c1nc2scnc2c(NC2CCc3cccnc32)[nH]1)N1CCC(C)C1 43070,C(C(O)C(=O)NC1(c2noc(C)n2)CC1)NC(CC1CC(NC)C1)=O 43071,C1(N(C)C(C2CCOCC2)=O)CCN(C(C2COCCN2CC(F)F)=O)C1(C)C 43072,CC(C)CC(CNC(C1CCN(C(C)C)C1)=O)NC(=O)CCCCNC(N)=O 43073,C1(CNC(CNC(C)=O)=O)CC2CC(C1)N(C(=O)CC1CC3CCC1CC3)C2 43074,C1(C(C)NC(=O)CN(C)CCO)CCCN(C(=O)CCCn2cccn2)C1 43075,C1(c2nnc(N(C)CC)n2CC2CCCO2)(Cn2nc(C)cc2Cl)CC=CCC1 43076,Cc1ncc(C(=O)NC2CC(OCC(=O)N(CC(C)(C)C)C(C)C)C2)c(=N)[nH]1 43077,Cc1noc(C)c1CCC(=O)NCCN(C(C1(C#N)CC1C(F)(F)F)=O)C1CC1 43078,c1ccc(C2CC(NCc3cnc(C4CCC4)o3)CN2)cc1 43079,CC1CC(C(N2CC(O)(CNC(=O)CSCC(F)F)C2)=O)CN1C 43080,c1(NC(C)=O)ncc(S(=O)(=O)N2CCCC(c3ccc(CO)cc3)C2)s1 43081,Cc1ccc(C2CC2C(=O)NCC2(F)CCC(NC(=O)Cc3c[nH]nc3O)C2)cc1 43082,c1(C(=O)NCC(=O)NCC2CC(NC(=O)CC3CCC4CC34)C2)ccccc1Cl 43083,C1(NCc2n(C)cc(Br)c2)CC2(CCCC2)C1 43084,C(C(CC(C)C)C(=O)NC12CC1CN(C(c1ccnc(C3CCC3)c1)=O)C2)OC 43085,CC1(C)C(=O)CC1C(N1CC(C(=O)NCC(C)(C)C2(O)CCC2)C(F)C1)=O 43086,C1(NC(c2cc(C)c(O)nn2)=O)CC2CCC(C1)N2C(=O)CC1CCC(=O)NC1 43087,C(C(CC(C)C)NC(=O)Cc1ccc(F)cn1)NC(C1CC(C)(CC)C1)=O 43088,C(C)(CC(C)NC(c1sccc1COC)=O)NC(CN(C)CC)=O 43089,N1(C(CC(CC(=O)OC)C)=O)CCN(C(C2CC(=O)N2)=O)CC(C)(F)C1 43090,CC1CCN(c2nnc(C(F)(F)F)s2)C(C)C1NC(C1CSC1)=O 43091,C1(C(N(C2CCN(C(c3cnco3)=O)CC2)CC)=O)C2C(=O)OCC12Br 43092,c1(C(=O)NCC(CC(C)C)NC(=O)C=CS(C)(=O)=O)cc2cc(F)ccc2o1 43093,c1(C(N2CC(NC(c3nccc(C)n3)=O)C3C2C3)=O)cc2cccnc2s1 43094,C(=O)(C(=O)C(F)(F)F)NC(C1CCN(C(=O)COc2cnn(C)c2)CC1)C 43095,C#Cc1cc(C(=O)NCCC(C)NC(C2(C)CCCS2(=O)=O)=O)ccc1C 43096,c1(C(N2CCC3(CC3C(N3CCC(O)CC3)=O)C2)=O)cc(Cl)cc(Cl)c1O 43097,CCCC(CCNC(C1CN(C)CCN1C(=O)CCC(N)=O)=O)CCC 43098,C1(NC(c2c(C)ccnn2)=O)COC2C(NC(=O)CCCC(F)F)COC12 43099,c1(CN(S(=O)(=O)CC2(C(N)=O)CCCCC2)CCC)c(Cl)nc2sccn12 43100,c1(Nc2nnc(C(C)OC)s2)nc(Cl)cc2cc(Br)ccc12 43101,Cc1cc(S(N)(=O)=O)sc1C(N1C(CNC(C2CC(F)C2)=O)CC2CC12)=O 43102,N1(C(C2CC(=C)C2)=O)CCC(CC)(NC(c2ccccn2)=O)CC1 43103,Cc1nc(C(N2CC3(NC(=O)CCC4CCC(O)CC4)CC2C3)=O)n(C)n1 43104,N1(CCSc2cn(C3CCC(C(=O)O)C3)nn2)CCN(c2ccnc(O)c2)CC1 43105,C12(NC(C(C)CC(F)F)=O)CCOCC1CN(C(=O)COc1cnc(Cl)cn1)C2 43106,C1(CNC2CC(C)SCC2)CCc2n[nH]cc2C1 43107,c1(CCC(=O)NCC2C(NC(C(CC)F)=O)COC2)ccc(Cl)cc1Cl 43108,O=c1cccnn1CCc1nc(Cc2ccoc2)no1 43109,Cc1ccc2c(c1)CN=C2NC(C1CC(F)(F)C12CCC2)=O 43110,C1(NC(C(C(=O)OC)C)=O)CN(C(c2cc(C)ccc2Cl)=O)CCC1(F)F 43111,c1(C(=O)NCCCC(C)(C)NC(C2CC3CC2CC3O)=O)ccc(C#N)cc1F 43112,c1(C(=O)OC)cc(NC(=O)NCCCC(c2ccccc2)C2CC2)c(Br)cc1C 43113,C12(CNC(=O)CC3CCOC3)CCC(CN(C(C3CCCCC3O)=O)C1)C2 43114,N1(C(c2n(CCC)ncc2)=O)CCC(C(=O)NCC(C)C)C1(C)C 43115,N1(C(CCCCC#C)=O)C(CNC(c2cnc(CC(C)C)[nH]2)=O)CC2CCCC12 43116,CCCCC(CNC(=O)C(C)NC(=O)NC)NC(c1cocc1C)=O 43117,CCCC(C(O)C(=O)NCC(F)(CC)CC)NC(=O)C(O)C(C)(C)C 43118,c1(C(=O)NCC2N(C(CCP(C)(C)=O)=O)CCC2)ccc(N)c(Cl)c1O 43119,CC(N=c1[nH]c(=NC2CCN(c3ncccn3)C2)[nH]c2c1COCC2)C1CCC1 43120,C1(C(N2CCCC(OC)C2)=O)COCCN(C(C2CC2(C)C(F)F)=O)C1 43121,Cc1nc(N2CCCC2)nc(O)c1CC(N1CCN(C(=O)CO)CC1C1CC1)=O 43122,N1(C(CCCC(=C)C)=O)CC2COCCC2(NC(C2CC2C(N)=O)=O)C1 43123,Cc1cc(N)c(C(=O)NCC2(CN(C(=O)CC3CC4(CC4)CO3)C)CC2)nc1C 43124,C1(NC(C(c2cccnc2)N(C(=O)Cc2csnn2)C)=O)CCC(C)(C)CC1 43125,CC(C)CC(C(=O)NC(C)CNC(c1ccncc1Cl)=O)N1CCCCC1=O 43126,c1(CC(=O)NCC2N(C(C3CCN(CC)CC3)=O)CC(O)C2)cccc(F)c1F 43127,c1(C(CNC(CC2CC(OCC)C2)=O)NC(c2ncn(C)n2)=O)ccc(F)cc1 43128,C1(N(C(=O)CCc2ncco2)CC)CCCN(C(=O)CCC2CCCO2)CC1 43129,c1(CC)n[nH]c(CC)c1CC(N1CC(C)(NC(C2CC2C)=O)C1)=O 43130,Cc1ccc(C(N2CCN(C3CCC(NC(c4cc[nH]c4)=O)C3)CC2)=O)cn1 43131,CC(C)C(CC(=O)N1CCN(C(c2cc(Cl)cs2)=O)CC1CO)c1ccccc1 43132,C(=O)(C(C#N)CC1CC1)NCC(CCC)NC(c1ncsc1C)=O 43133,CCC(CNC(=O)Cc1ccc(CO)cc1)(CC)NC(=O)C=Cc1scnc1C 43134,c1(C(=O)NC2C(CNC(c3cc(OC)ncc3)=O)CCC2)noc2c1COCC2 43135,N1(C(CC(C)C)=O)CCC(N(C)C(c2cc(-c3cccnc3)[nH]n2)=O)C(C)C1 43136,N1(C(C=C(CC)C)=O)CCC2(NC(=O)Cc3c(F)cccc3Br)CC2C1 43137,C12CCC3(CN(C3)C1=O)O2.Cc1cc(C(=O)NCCOCc2cccnc2)c[nH]1 43138,C1(CC(=O)NC2CC(F)(F)CC2NC(C2SCCCS2)=O)CN2CCC1CC2 43139,N1(C(COc2c(C)cccc2Br)=O)CC2(CCN(C(C3CC(C)C3)=O)C2)C1 43140,c1(C(N2C(CNC(C3(C(C)(F)F)CC3)=O)CCC(C)C2)=O)cnn2c1OCCC2 43141,c1(C(=O)NCC2CCN(C(C3(C#C)CCCC3)=O)C2)cnn2c1CC(F)(F)C2 43142,Cc1cccc(CN(C(C)=O)CC2CCN(C(C3CCCCO3)=O)CC2)c1 43143,N1(C(C(C)(C)OC)=O)CCN(C2CCCN(C(c3cnsn3)=O)C2)C(=O)C1 43144,N1(C(c2c(C)scn2)=O)CCC(OCCNC(=O)CC2CCS(=O)(=O)C2)CC1 43145,CC1=CCC(C(=O)NCCCN(C(=O)CC(C)NC(=O)OC(C)(C)C)C)CC1 43146,CCCC(O)C(CO)NC(C1(CN(C)C)CCC1)=O.C12(CC1)C(=O)N2 43147,N1(C(c2n(C)ncc2)=O)CC(C(N2CCCC3C(O)CC23)=O)CCC1(C)C 43148,C1(COC)(NC(=O)NC2CCCCC2OC)CC(C)(C)C1 43149,N1(C(COC)=O)CCC(CNC(C2CC3CCCCN3C2)=O)C(F)(F)CC1 43150,C(=O)(CC(O)CCCC)N(CCCCC(N1C(CC=C)CCCC1)=O)C(C)C 43151,Cc1cc(CCC(=O)NCCC(O)CNC(C2(C)CCN(C)C2=O)=O)cc(C)c1 43152,C#Cc1cncc(C(=O)NCCC2CC(F)(F)CN2C(c2nocc2Cl)=O)c1 43153,CC1CN(C(c2cc(OCC3CC3)ncc2Cl)=O)CCN1C1CCCCC1 43154,C(CC(C)CC)(C(=O)N1C2COCC1C2)NC(CC=C=C)=O 43155,n1(CC(N2CCC(CNC(C(C(C)C)OC)=O)CC2C)=O)cc([N+](=O)[O-])nc1C 43156,N(C1CC(C)n2ncnc21)C(C1CCC(NC(C2(C=C)CCC2)=O)CC1)=O 43157,N1(C(c2c(N)nc(Br)cc2)=O)CCC2(C1)CN(C(C1CCC(O)CC1)=O)C2 43158,N1(C(c2n(C)cnc2)=O)CCC(C)(C)C(C(=O)NCC2CCC(F)(F)C2)C1 43159,c1(C(=O)NC(C(C)C)CCNC(=O)C(C)(C)C)nnc2n1CCCC2 43160,C1(NC(C2(CCCC)CCC2)=O)CN(C(C2CN(C)C2)=O)C2(CCOC2)C1 43161,C1(CNC(c2cc(F)c(F)c(F)c2)=O)CC2(CCN(C(=O)C(Cl)=CCl)CC2)C1 43162,CCC(C)(C)CCCC(=O)NCCC(C)NC(c1nc(C)ncc1Br)=O 43163,CC(C)(CC(=O)N1CCC(O)(CNC(=O)CCCC(F)(F)CO)C1)CC(F)(F)F 43164,c1(C(=O)NCC#CCNC(=O)CCc2cnccn2)cc(Cl)c2c(c1)OCO2 43165,C(=O)(C(F)(CNC(=O)C(C1CC1)C1CC1)C(C)C)N(CC)CC1CCCOC1 43166,c1(C(N2CC(C)C(C)C2)=O)cc(Br)cc(F)c1N 43167,N1(C(Cc2cc(C)[nH]n2)=O)CC(C)(C(=O)N(CC2=CCSC2)C)CC1(C)C 43168,C(=O)(CC(C)(C)C(F)F)N(CC(C)(C)CNC(=O)Cc1ccon1)C 43169,C1(CC=C)(NC(C2CCSC(C)C2)=O)CCCN(C(c2csc(C(C)=O)n2)=O)C1 43170,c1(C(C)NC(C(=CC2CCC(C)CC2)C)=O)cnn2ccccc12 43171,C1(CC(N2CC(NC(C(C)OCC#C)=O)(CO)C2)=O)COCC(C)(C)O1 43172,N1(CC(C)(C)C)CCC(F)(F)C(CNC(=O)CC(=O)N(C)C)C1 43173,N1(C(Cc2c(C)cnn2C)=O)CC(C)N(C(=O)Cc2ccoc2C)C(C)C1 43174,O(NC(=O)C(CNC(=O)C(c1cccnc1)O)CC(C)C)Cc1ccc(C)cc1 43175,N1(C(C(C2CC2)SC)=O)CCC(C)(NC(=O)CC2(O)CCCCC2)CC1 43176,C1(NC(CCCCSC)=O)CCC2(CC1)CC2NC(=O)C(=O)N(C)C 43177,CC1CCN(C(c2cnc(N)c(Br)c2)=O)CC1NC(=O)C(C)(C)C1CC1 43178,N1(CC(=O)N(CC(=O)N(CCCCO)C)C)CCC(=O)CC1 43179,C1(C(=O)NCC=CCNC(C2(COCC)CC=CC2)=O)CC(C2CC2)C1 43180,C(=O)(C(CCNC(=O)CCn1cncn1)OC)N1CCC(C(CC)CC)C1 43181,c1(C(=O)NCC(Cc2ccccc2)N(C(C2CC(=C)C2)=O)C)ccn(O)c(=O)c1 43182,CC1CN(C(=O)CC2CC3CCC2O3)CCC1CNC(C1(O)CCCCCC1)=O 43183,c1(C(C(=O)NC2(C)CC2)N(C(c2ccccc2)C(=O)OC)C)c(SC)cccc1F 43184,C12(NC(CCC=CC(C)C)=O)CCC1CN(C(C1(N(C)C)CC1)=O)C2 43185,c1(C(N2CCC3CN(C(C4ON=C(C)C4)=O)C3C2)=O)cnc2sc(C)cn2c1=O 43186,c1(C(=O)NC2CN(Cc3cnc(Cl)cn3)CC2F)cc(F)c(F)cc1F 43187,C1(NC(CC2(C)N(C(c3c(CC)n[nH]c3)=O)CC2)=O)CC2OC(=O)CC12 43188,C1(N(C)C(C2CC2C(N)=O)=O)CCC(NC(c2c[nH]nc2C(C)(C)C)=O)C1 43189,C=CCC(C)(O)C(=O)NC1CN(C(c2cnon2)=O)C1 43190,C1(C(=O)NCCCN(C)C)Cc2c([nH]c3ccccc23)CN1C(c1ccon1)=O 43191,c1(SC)cc(F)ccc1NC(=O)NC(C)Cc1ccc(NC(=O)C(C)(C)C)cc1 43192,c1(SCC(=O)NC2COCCN(C(CC(=O)OC)=O)C2)ccc2c(c1)CCC2 43193,N1(C(c2c(C)ncc(C)c2)=O)CCN(C(=O)CC(O)C(C)C)C2(CCC2)C1 43194,N1(C(C(CC)(C)OC)=O)CCCN(C(=O)CCNC(c2ccc(C)cc2)=O)CC1 43195,C1(NC(CC2CCN(C(C(C)OCC3CC3)=O)CC2)=O)CN(C)CCN(C)C1 43196,N1(C(C=C(CC)C)=O)CC(CNC(=O)Cc2cc(-c3ccccc3)on2)C2CC12 43197,C#Cc1ccc(OCC(=O)NCCC2CN(C(c3conc3C)=O)C2)cc1 43198,c1(C(N(CCN(C(C2C(C(=O)OC)C2)=O)C)C)=O)nnn2c1CSCC2 43199,C(CCCCC(=O)NC(C)CCC(=O)NCCCc1ccncc1)=CC 43200,C(C)(CCCN=c1nc(C(F)(F)F)c2ncccc2[nH]1)OC 43201,C=CC(C)C(C)C(=O)NCC1(NC(=O)CC2CS(=O)(=O)C2)CCCC1 43202,c1(C(=O)Nc2cncc(C(=O)OCC)c2)cc(Br)cc2c1cnn2C1CCCC1 43203,CC1CN(C(C2CC2c2cccc(Cl)c2)=O)CC1NC(=O)C(C)(F)F 43204,c1(C(N2CCN(C(C(=O)NCCC)C)CC2)C)nccc2ccccc12 43205,C#Cc1cc(C(=O)NC2C3CC(NC(C4CCC(OC)C4)=O)CC23)ccc1C 43206,c1(CC(=O)NC2CCN(C(C3(c4ccon4)CCC3)=O)C2)ccccc1OCCF 43207,C(=O)(N=c1cc[nH]cc1SC)C1CCC2(CN(C(C(CCC)O)=O)C2)O1 43208,c1(OC)cnc(N2CCN(C(=O)NCC(N3CCOCC3)(C)C)CC2)nc1 43209,N1(C(c2n(CC#C)ccc2)=O)CC(NC(=O)C(C)c2cc[nH]n2)CCC1C 43210,C(c1c(N)cnn1C)=CC(=O)N(CC(C)CNC(C1CCCC1C(F)(F)F)=O)C 43211,c1(C(N2C3C(NC(CC(C)F)=O)(CCC3)CC2)=O)nn(C)c2c1CCCC2 43212,Cc1oc(C(C)C)nc1C(=O)NCC(C)NC(=O)CC1CC(C(F)F)C1 43213,CC(C)C(C)CNC(=O)C(C)N(C(=O)CCCNC(N)=O)C 43214,c1(N2CC(C)S(=O)CC2)ccc(S(=O)(=O)NCCc2cnoc2)cc1Cl 43215,CC(C)CC(O)C(C)C(=O)NCc1ccc2ccccc2c1 43216,N1(C(C2C(CC)OCC2)=O)CCC(CCNC(C2(OC(C)=O)CCCC2)=O)CC1 43217,c1(CC)cccnc1C(=O)NCCC1(O)CCN(C(=O)C(C)OCCC(C)C)C1 43218,c1(C(N2CCN(C(c3c(C)ccnc3O)=O)CC2C)=O)cccc(C#N)c1Br 43219,O=S(=O)(c1c[nH]ccc1=NCC1(F)COCCOC1)NCCC1CCCCCCC1 43220,c1(C(=O)NCC2N(C(c3c(C)nccc3)=O)CC2)nnc(O)c(Br)c1O 43221,c1(OC)cc(C(N2CCC(NC(C3(C)CCC(=O)N3)=O)C2)=O)sc1S(N)(=O)=O 43222,C(CNC(=O)C(C)CN(C)C)(CC(F)(F)F)NC(C=Cc1nnc(C(C)C)o1)=O 43223,c1(CNC2CCC(C(=O)Nc3cc(OC)n[nH]3)C2)c(F)cc(Br)c(F)c1F 43224,CCCS(=O)(=O)C(C)C(=O)NCc1cc2ccccc2s1 43225,c1(C(N(C2CCN(C(C3=C(C)CCC3)=O)C2)CCO)=O)c(C)nn2c1CCCC2 43226,S(=O)(=O)(c1cccc(=NC(C)C2CCCCO2)[nH]1)NCC(C)C1CCC1 43227,CCCN(OC)C(=O)CC1CCN1C(c1cn(CC2CC2)nn1)=O 43228,C12CN(CC1C(=O)O)C2=O.c1(CN(C(CC)C(=O)O)C)ccc(C(N)=O)cc1 43229,N1(C(c2c(OC)ncc(C)n2)=O)CCc2cc(-c3ccccc3CO)ccc2C1 43230,C1(C(N2CCC(C(C)NC(=O)C(c3cccnc3)O)CC2)=O)CCCCC(=O)C1 43231,c1(C(=O)NCC(CNC(C=CC(=O)NC2CC2)=O)F)ncoc1C1CCCO1 43232,C1(C(=O)NC(c2ccccc2)CC)CCC(n2cc(C3CCC3)nn2)C1 43233,CCCC(C)CC(=O)NCCOCCCNC(=O)CC=C(Cl)Cl 43234,CC1CC(NC(C2(C)CCN2C(=O)C=Cc2ccncc2)=O)c2nccn21 43235,N1(C(=O)OC(C)(C)C)CCC2CCCC12COC(=O)Cc1cncnc1O 43236,CC(C)C(C(C)NC(C12CCN(CC1)C2)=O)NC(c1cc(C(F)(F)F)n[nH]1)=O 43237,C12(CNC(=O)Cn3nnnc3C3CC3)CCC1CN(C(C1C=CCCC1)=O)C2 43238,C(=O)(C(F)C(C)C(F)(F)F)NC1C(CC)CN(C(=O)C=Cc2cn(C)nn2)CC1 43239,Cc1cncc(C(=O)NC2CC(NC(c3cn(C4CC4)cn3)=O)C2)c1 43240,c1(NC(=O)NCCc2ccn(C)n2)cc(Nc2ncc(F)cn2)cc(Br)c1 43241,c1(C(=O)NC(CN(C)C)C(=O)NCC#CC(F)(F)F)ccc(C#N)n1C 43242,C1(NC(CN2C(C)CCC2)=O)C=CCN(C(c2ccc(O)nn2)=O)C1 43243,Cc1ncc(C(=O)NCC2C3CN(C(=O)C(O)CC(F)F)CC23)c(C2CC2)n1 43244,c1(C(=O)NCC2N(C(C(CCOC)OC)=O)CC(OC)C2)scc2c1CCCC2 43245,C(C(C)(C)CNC(=O)COC1CC1(F)F)N(C(C1C(C(=O)NCC#C)C1)=O)C 43246,C1(C(=O)NCC#CCCO)(CC)CCN(C(=O)C(C2(O)CCCC2)F)CC1 43247,C1(NC(c2c(CC)ncnc2)=O)CN(C(=O)Cc2cccc(F)c2)C2CCCC12 43248,C1(c2n(CC(=C)C)nnn2)(NCC2(F)CC(C(N)=O)C2)CCOCCC1C 43249,N=c1[nH]c(=NC(CCO)c2ccc(F)cc2F)[nH]c(=NC2CCC(=O)NC2)[nH]1 43250,c1(C(=O)NC(C(C)NC(Cn2c(C)cnc2)=O)C)ccc(C(N)=O)c(Cl)c1 43251,C1(C(=O)NC2CCN(CC)CC2)CCCN(C(=O)CC2CCCO2)C1C 43252,CC1CC(O)CCN(C(=O)CC(C2CC2)NC(c2cnn[nH]2)=O)C1 43253,C(CCCC(CO)NC(=O)C(F)C1CCC1)NC(c1ncn(C(C)C)n1)=O 43254,C1(NC(C(C)NS(C)(=O)=O)=O)CC(NC(=O)CCc2csc(=N)[nH]2)CC1O 43255,c1(C(=O)NCC=CCNC(c2cscn2)=O)cc(C2CC2)[nH]n1 43256,C1(C(CCC)C)CCCCN1N1CCC(CCOC)(C(=O)OCC)CC1 43257,N1(C(C(C)N(C(C(COC)C)=O)C)=O)CCC12CC(CO)C2 43258,c1(C(=O)Nc2c(C#N)ncc(Br)c2)ccc2cccc(-c3cnoc3)c2n1 43259,C1(C(=O)NCCC2C=CCC2)(N(C(C(C)N2CCCC2)=O)C2CC2)CCN(C)C1 43260,N(C(=NCCN(C)Cc1ccc(Br)cc1)NC1CCOCC1)C1CCC(SC)C1 43261,c1(C(N2C(CCNC(c3ccc(C)s3)=O)CC(OC)C2)=O)cccn2cnnc12 43262,c1(C(=O)NCC=CCNC(CC)=O)ccc(=O)n(CCF)n1.C12(CO)CN(C1)C2 43263,C(=O)(CC(C)C(F)(F)F)NCCCC(C)NC(C(C(C)C)C)=O 43264,C1(NC(C(C)OCC)=O)CS(=O)(=O)C12CCN(C(c1cc(Cl)nc(=N)[nH]1)=O)CC2 43265,FCCCN=C(NCC1(c2ccc(F)cc2)CCCC1)NC1CC1C1CCCO1 43266,C(=O)(CCC(=O)N1CC=CC1CNC(=O)C(O)CC1CCOCC1)OC 43267,C1(C(=O)NCCN(C(=O)C(C)n2cnnn2)CCOC)(OCC)CCOC1 43268,N1(C(CC(C)c2ccccc2)=O)CCN(C(=O)COCCOCCO)C2CCC12 43269,c1(C(N2CCC2Cn2cc(CC3CCOCC3)nn2)=O)cc2n(c1)CCCC2 43270,c1(N2CCC(N(C34CCCCC3C4)CC)CC2)nc2ccc(C)nc2s1 43271,C1(C(N(C(C)CNC(c2ccccc2SC)=O)CC)=O)NC(=O)OC1C 43272,N1(C(c2occ(C)c2)=O)CCC2(CC1)C(NC(C1(C3CCC3)CC1)=O)CS2(=O)=O 43273,Cc1cc(C(=O)NC2CC2NC(=O)C(C2CCCCC2)C)cnc1C 43274,c1(CNCC2N(C(CN(C3CCCN3C)C(C)=O)=O)CC=C2)ccc(F)c(F)c1 43275,Cc1cc(C)c(C(=O)NC23CC2CN(C(=O)C=C2CCCCC2(C)C)C3)c(=O)o1 43276,c1(CNC(C2N(C(C)(C)C)CC2)=O)cnn2c1CN(C(C1CC1C(N)=O)=O)CC2 43277,c1(-c2ncc(C(N(CC(c3ccncc3)O)C)=O)s2)cccc(Cl)c1 43278,N1(C(C(N2C(CC)CCC2)=O)=O)CCOCC1CNC(=O)Cn1nc(C)cc1C 43279,c1(-c2nc(-c3cn(C)[nH]c3=N)on2)cccc(S(=O)(=O)CCO)c1 43280,N1(C(C(n2cc(-c3ccc(N)cc3Cl)nn2)C)=O)CCc2cnccc2C1 43281,c1(N2CCN(c3cc(NC(CC=C)C(=O)O)ncn3)CC2)c(F)ccc(Cl)c1F 43282,C(CS(=O)(=O)CC(=O)N1CC2(CC(NC(=O)CCCCC(C)C)C2)C1)OC 43283,c1(C(=O)NCC2CCCN2C(C2CCS(=O)(=O)CC2)=O)ccc2ocnc2c1 43284,N1(C(CC=C)=O)Cc2[nH]nc(C(=O)NCC(COC)C(C)C)c2C1 43285,N1(C(c2c(C)n[nH]c2C)=O)CCCC1C1CCCN1C(c1csnc1Cl)=O 43286,Cc1c(NC(=O)CN(c2ccc(C#N)cn2)C)cc(F)cc1[N+](=O)[O-] 43287,N1(C(c2c(CC)csc2)=O)CCC2(CCN(C(=O)COC)C2)C1 43288,C(=O)(C(C)(C)CC(C)(C)C)NC1CC(C)N(C(C2CCSC(C)C2)=O)C1 43289,Cc1cc(C(=O)NC2C3CC2CN(C(=O)C(C)C(C)C)C3)c(N)c(C)c1 43290,c1(C(N2CC(CC)N(C(=O)C(O)CC(C)C)CC2)=O)ccc2ocnc2n1 43291,CC(C)CC(C)(O)C(=O)N(C)CC1CCCN(C(c2cc(C(F)(F)F)c[nH]2)=O)C1 43292,C1(C(N(CCNC(C2(C(F)(F)F)CCN(C)C2)=O)CC)=O)CNC(=O)CC1(C)C 43293,c1(NC(C(CCN(C)C)NC(=O)C(O)C2CC2)=O)ccc2nccn2c1 43294,C1(CC)CN(C(=O)Cc2ccc(C(F)F)cc2)CCN1C(c1ncc(F)cn1)=O 43295,C1(N(C(C=C(CC)CC)=O)C)CN(C(=O)C(C)C2CC2)CC1(C)C 43296,C(CCC(C)(C)C(=O)NCc1nonc1C)NC(C(=Cc1ccco1)C)=O 43297,C=CCC(CC(=O)Nc1cnc(Cl)cc1C)NC(=O)CCC1OCCO1 43298,c1(C(=O)NC(C(N2C(C(CC)C)CCC2)=O)C2(O)CC2)cnn2c1CCC2 43299,N1(C(C2C(OC)CCC2)=O)CCCC2CN(c3ncc(O)cn3)CC12 43300,C1(C(N2CC3C(C(=O)NC(CC(=O)NC)C)C3C2)=O)CC(=O)NC(C)C1 43301,C#CCC(CC(=O)NC(C(C)C)C1CCC1)NC(=O)CCCNC(C)=O 43302,c1(NC)cnccc1C(N1CCC(CF)(NC(c2ccco2)=O)C1)=O 43303,C(C(C)C(C)C(=O)NC1CC(F)(CNC(=O)COCc2ccnc(O)c2)C1)OC 43304,c1(CC(=O)NC2CCC2NC(c2ccc(O)nc2Cl)=O)n[nH]c2ccccc12 43305,N1(C(COC2(C)CN(N(c3ccc(C=O)o3)C)C2)=O)CCCC1(C)C1CC1 43306,C(=O)(NN1CCCC1C(=O)NCC(C)(CO)OC)c1cc(CC)nn1C 43307,Cc1sc(Cl)nc1C(N1CC(NC(c2cc(C(N)=O)c[nH]2)=O)CC1C)=O 43308,C1(C(N(CC(=O)NCCC)C)=O)N(C(=O)C(C)SC(C)C)CCC1(C)C 43309,Cc1ncnc(C)c1NC(C1CCCCN(C(C23CC(F)(C2)C3)=O)C1)=O 43310,N1(C(C(C)CS(C)(=O)=O)=O)CCN(C(=O)C=CCn2cncn2)C2(CCC2)C1 43311,N1(C(C=C(CC)CC)=O)CCC(O)(CCNC(c2csc(Cl)n2)=O)CC1 43312,C(c1cncc(C)c1)=CC(=O)NC(CC)CNC(=O)CSCc1ncc[nH]1 43313,c1(C(C(=O)NC)C(N2CCC2C2CCC2)=O)ccc(OC(F)(F)F)cc1 43314,CCCC(CCCS(C)(=O)=O)C(=O)NCCCC(C)NC(=O)CC1(C)CCCC1 43315,c1(C(N2CCC(NC(C3(C)CCC(C)CC3)=O)C(O)C2)=O)c(F)cc(Cl)cc1F 43316,c1(C(=O)NC2CN(C(c3c(OC(C)C)cccc3)=O)CC2O)cc(Cl)ccc1Cl 43317,c1(C(=O)NC(CCNC(C2(C(C)C)COC2)=O)C)cc(C(N)=O)cs1 43318,C1(C(N2C(CC#C)CCCC2)=O)CN(C(=O)CCc2cnn[nH]2)CCN1C 43319,c1(C(N(C2CCN(C(C3CC3[N+](=O)[O-])=O)CC2)C)=O)cnc2c(c1)C(=O)CCC2 43320,Cc1cc(C)n2nc(C(=O)NCCCCC(C)NC(=O)Cc3cnco3)nc2n1 43321,N1(C(C(C(C)C)SCC)=O)CCN(C(=O)Cc2sc(C)nc2C)CC(C)(C)C1 43322,C(=O)(CCC(C)(F)F)NCC(C)C(=O)NCCN1CC(C)(O)C1 43323,N1(C(C(C=C)(C)CC)=O)CC(C2CN(C(c3[nH]c(=N)ccc3C)=O)C2)C1 43324,c1(N2C(C(=O)OC(C)(C)C)C3C=CC2C3)ncnc2[nH]c(I)cc12 43325,N1(C(Cn2ncc(C)c2)=O)CCCCC1c1cn(Cc2ccoc2C(=O)O)nn1 43326,C(CC)(CCCC(=O)NCc1cc(C#N)cs1)NC(C1(CC#C)CC1)=O 43327,C(CCC(N)=O)(C(=O)NCC(C)(CO)NC(=O)Cn1nnc(=N)[nH]1)N(C)C 43328,CCCCC(CC)C(=O)NC(C)(C)C(C)NC(=O)C(=O)Nc1ccc(CC)cc1 43329,C1(C)(CNC(CCN(CC=C)C(c2cc(N)cc(F)c2)=O)=O)CCCCC1O 43330,C(CCC(C)C(=O)NCC1(C)CCN(C(C2(C)CC3CCC2C3)=O)CC1)OC 43331,C(=O)(C1Cc2ccccc21)N1CCCC(CCCCNC(c2occ(C)c2)=O)C1 43332,c1(C(=O)NCC(CC)NC(c2ccn(C)c(=O)c2)=O)cnc2ccc(C)cc2c1 43333,c1(C(=O)NCC2CC2CNC(c2n[nH]cc2C2CCC2)=O)csc(Cl)n1 43334,Cc1nc(N2CCC(C)C2CNC(C2COCCN2CC(F)F)=O)[nH]c(=N)n1 43335,c1(C(=O)NCC=CCNC(C(C2CC2)SC)=O)cccc(CS(C)(=O)=O)c1 43336,C1(C(N2CCC(C)(CNC(c3c[nH]c(=NC)s3)=O)C2)=O)CCN(C2CC2)S1(=O)=O 43337,c1(C(N2CCC(C)C(NC(C3(C)CC(C#N)C3)=O)C2)=O)ccc(Cl)c2occc12 43338,n1(CC)cc(Cl)c(C(N2CCCC2C(C)(C)NC(=O)C(COC)N(C)C)=O)n1 43339,c1(C(N(C(CNC(CCOC(C)C)=O)C)C)=O)ccc(F)cc1 43340,C1(N(C(=O)COCC2CC2)CC#C)CCN(C(c2cc(O)cs2)=O)CC1 43341,c1(OCC)cccc(C(=O)OCc2ccc(OC)nc2F)c1CSc1ccccc1 43342,N1(C(C2(CC)CCCO2)=O)CCCC(N(C(=O)CCC2OCCO2)CCO)C1 43343,C(=O)(C(C)C(C)C(C)(C)C)NCCC1(CNC(c2c(C)cc(CC)o2)=O)CC1 43344,C(C)(C)(CC(=O)NCC(O)CC(=O)Nc1c(C)noc1C)OC 43345,N1(C(c2c(CC)n[nH]c2)=O)CC(C(N2CCC3C(OC)CC23)=O)C(F)(F)C1 43346,C(C(C)(C)C(=O)NCCC1CN(C(=O)C(C)Cn2ccnc2)C1)OC 43347,c1(NC(C(N2CCN(C3COC3)CC2)C)=O)ccc(C2CCC(=O)N2)cc1 43348,C1(CNC(c2cc(-c3ccc(C)s3)[nH]n2)=O)CCC(C)CN1C(=O)C(N)=O 43349,Cc1cc(O)cc(C)c1CC(=O)NCC1(O)CC(NC(c2cc(CO)[nH]n2)=O)C1 43350,c1(C(N2CC(NC(C(COC)C)=O)C2)=O)ccc(N2CCOC2=O)cc1 43351,Cc1ccc(C(N2CCCCC2CNC(=O)C(C)(C)C(N)=O)=O)c(O)n1 43352,c1(C(N2CCC(C(=O)NCC=C3CCSCC3)(OC)C2)=O)cc(C#N)oc1C 43353,C1(C(=O)NCCOCCN(C)C(c2cccs2)=O)CCCC1S(C)(=O)=O 43354,C1(CNC(c2ccc(=O)n(C3CC3)c2)=O)CC(F)(F)CN1C(c1scnc1Cl)=O 43355,N1(C(CCOC2CN(C(CC3CCC(C)CC3)=O)C2)=O)CCCNC(=O)C1C 43356,C1(C(=O)NC2C3CN(C(CN(C)C4CC4)=O)C2CC3)CCn2cnnc2C1 43357,C=CCC(C)C(=O)N1CCC(OCCNC(C2C(C(=O)OC)C2(C)C)=O)C1 43358,c1(CC(N2C(CN(C(CNC(CNC(C)=O)=O)=O)C)CCC2)=O)ccnc(O)c1 43359,N1(C(C(CCC)NC(C)=O)=O)CC(C2CCCN(C(=O)C(C)CS(C)(=O)=O)C2)C1 43360,C1(C)(CNC(Cn2c(C)c(Cl)cn2)=O)CN(C(c2cncnc2)=O)CCO1 43361,Cc1cccn2cc(CC(=O)NC3COCC3NC(=O)Cc3csc(Cl)n3)nc12 43362,c1(C(N2CCCC(CCC)(NC(=O)C(O)C3CCC3)C2)=O)ccc2nncn2c1 43363,C1(F)(C(=O)NC(C(=O)NC(C)CCC2CC2)C)CCCCC1.CCS 43364,C12(CNC(C(CC)c3ccccc3)=O)CC(NC(c3cc(C)[nH]n3)=O)(CCO1)C2 43365,c1(C(C)(C)C)ccc(C(=O)NC2CC(NC(C3CC3(F)F)=O)C2)o1 43366,C1(CC(=O)N(C)CC=CC(=O)NC(C)(C)CC2CCOC2)CCCC1C1CC1 43367,c1(C(N(CCCCNC(CC2CCN(C)C2)=O)C)=O)cncc2nc[nH]c12 43368,c1(C(=O)NC2CN(C(c3cnn(C4CC4(F)F)c3)=O)CC2F)c(F)cccc1Br 43369,c1(N2CCCC(C(C)C)C2)nc(N2CCS(=O)C3(CCC3)C2)nc2cccnc12 43370,C1(NC(c2c(C)cc(C)s2)=O)CN(C(C2CC3(C2)CC3F)=O)CC2(CCC2)C1 43371,c1(C2CCN(C(C=C(C)CCc3ccccc3)=O)C2)nc(C)cc(O)n1 43372,C1(CNC(C(C)c2ccsc2)=O)C2CCC1CN(C(c1cnc3[nH]cnc3c1)=O)C2 43373,c1(CC)cc(N)ccc1C(=O)NCC1CCN1C(C12CC(CO)(C1)OC2C)=O 43374,c1(C(N2CCOCC(NC(CC(C)(C)SC)=O)C2)=O)cc2cc(F)cc(F)c2[nH]1 43375,c1(-c2nc(COCc3nc(C)sc3)on2)cc(Br)cn2ccnc12 43376,n1(C(CC)CC)nc(C)cc1C(=O)NCC(C(C)C)NC(C1CCN(C)C1C)=O 43377,C1(CNC(C(CC)(F)F)=O)CC2CCC1N(C(=O)C(COC)NC(C)=O)C2 43378,CC(C)(CNC(C1(C)CCCN1C(=O)CCN1CCOC1=O)=O)C(N)=O 43379,C(=O)(C1=C(C)CCCC1)NC1C(SC)CN(C(=O)C(=Cc2ccc(F)cc2)C)C1 43380,C(C(CNC(=O)CCCOC(C)=O)C(F)(F)F)NC(C1CCN(CC)C1)=O 43381,c1(OC)c(C(=O)NCC#CCNC(C2CNC(=O)CC2C)=O)oc2ccccc12 43382,c1(CC)cc(C(=O)NC(CC(=O)NCC(=O)OC)C2CC2)n[nH]1 43383,c1(NC(C(C)SCc2nncn2C)=O)ccc(CNC(=O)C2=C(Cl)CC2)cc1 43384,n1(CC)nc(C(=O)NC(C)(CSC)C(=O)NCC(=O)OC(C)C)c(C)n1 43385,c1(OC)ccccc1CCCNC(=O)C(=O)NC1CCCNCC1 43386,c1(C(=O)NC(C2(C)CC2)C)ccc(CNN)cc1.C1(C(=O)O)CC1C 43387,N1(C(CC2N(C)CCC2)=O)CCN(C(=O)CC2(N(C)C)COC2)CC1CC(F)F 43388,N(C(=NCCC(C)=O)NC(C1(O)CCOCC1)C)Cc1cnn(CC)n1 43389,CCC(O)(C(=O)NCC(O)CN(C)C(C1(CC(C)C)CCC1)=O)c1ccccc1 43390,C1(C(=O)NCC2CC(NC(c3c(Cl)nc(OC)s3)=O)C2)CCCC2(CCC2)C1 43391,C1(CCNC(C(C)OCCC(C)C)=O)CCC(NC(=O)CCOC(C)C)C1 43392,CC(C)(CC(F)F)C(=O)NC1CC2CC1N(C(=O)CCc1ccc[nH]1)C2 43393,c1(OC)c(C(=O)Nc2ccc(C(=O)NCc3ccc(I)cc3)cn2)cccc1Br 43394,C1(CS(=O)(=O)Nc2ccc(C(=O)OCCOC)cn2)(OC)CCOCC1 43395,N1(C(c2ccn(CC)c(=O)c2)=O)CCCC2CN(C(C3(CC4CC4)CC3)=O)CC12 43396,c1(C(=O)NCC(=C)Cl)cccc2c(I)n[nH]c12 43397,Cc1cccnc1CC(=O)NCC1CCN1C(=O)CC1(c2ccon2)CC1CO 43398,C1(C(=O)NC(CCN(C(c2c(C)onc2)=O)C)C(C)C)CCC(=O)C(C)C1 43399,C12(C(=O)NC(CN(C(C(C)=CC3CC3)=O)C)(CO)CO)CC3CC1C2C3(F)F 43400,Cc1cc(C(F)(F)F)nn1CC(N1CC2CC2(CNC(C2C3COCC23)=O)C1)=O 43401,N1(C(=O)NC2(c3ccccc3Cl)CCC2)CC23CCCC2(COC3)C1 43402,c1(C(N2C3CCC(NC(c4cc5n(n4)CCC5)=O)(C3)C2)=O)nnn2c1CCCC2 43403,Cc1cc(NC(C2CC(F)CN(C(c3cc(Cl)cnc3Br)=O)C2)=O)cnc1C#N 43404,Cc1c(NC(c2csc(C3CC3)n2)C)ncnc1N1CCOC(C(N)=O)C1 43405,Cc1cccc(OCC(=O)N(C(C)CNC(C2(S(C)(=O)=O)CC2)=O)C)c1F 43406,Cc1c(N(CCCNC2CCCC2)C)ncnc1N1CCOC(C(C)(C)C)CC1 43407,c1(CNc2cc(N3CCOCC(C(C)N(C)C)C3)ncn2)cnc2sccn12 43408,N1(C(C(CC#C)CC(F)F)=O)CCCC2C1CCCN2C(=O)OC(C)(C)C 43409,c1(OC(CC)C)ccccc1C(=O)NC1CCN(C(=O)C(C)c2cccs2)CC1 43410,CC(C)CC(O)C(C)C(=O)N1CCC(CNC(c2coc(CO)c2)=O)CC1 43411,C1(C(=O)NC2C(NC(COC3(C#C)COC3)=O)C2)CN2CCCC2CO1 43412,CC(N=c1[nH]c(=NCC(CO)C(F)(F)F)c2[nH]ccc2[nH]1)c1c(F)cccc1Cl 43413,c1(OC)cc(CC(N2CC3CC(N(C(=O)C(C)C)C)C2C3)=O)cc(OC)c1O 43414,C1(CNC(=O)COc2ccccc2)CCN(C(=O)CSC(F)F)C12CC2 43415,c1(NC(C(N2C(C)CC(NC(C3(SCC)CC3)=O)C2)=O)=O)ccc(C)c(C)c1 43416,CCCC(C(=O)N1CC(C(=O)NCC2CCC2C)C1)OC 43417,Cc1cc(C(=O)NCCN2CCC(NC(=O)CC3CCC(=O)N3C)CC2)nn1C 43418,C1(C(N(CCC(=O)NCc2c[nH]nc2C(C)C)CC)=O)CNC(=O)CC1C 43419,c1(OC)ccccc1C1CC1C(=O)N(CC(C)(C)NC(c1nn(C)cc1C)=O)C 43420,N1(C(CC2CCN(C(C)=O)CC2)=O)CCOC2CN(c3nccc(C)n3)CC12 43421,n1(CC)nc(C(=O)N(CCCC(=O)NCC(C2CCCC2)C)C)c(C)n1 43422,c1(C(=O)NCC23C(CN(C(C(CC)SC)=O)C2)C3)ccc(F)c(C(C)C)c1 43423,C1(C(N2CC(C)(NC(c3cc(OCC)n[nH]3)=O)C2)=O)(C(=O)O)CC1S(C)(=O)=O 43424,c1(OC)cc2[nH]ncc2cc1C(N1CCC1C(=O)Nc1[nH]nc2cnccc12)=O 43425,C1(CNC(c2cnc(OC)s2)=O)CC2CCC1N2C(C1CN(C)C(=O)N1)=O 43426,C1(C(N2CC3C(NC(Cc4c(C)cc(F)cc4)=O)(C3)C2)=O)CN(CP(C)(C)=O)C1 43427,n1(CCOC)cc(C(N2CC(NC(=O)Cc3cncs3)CC(C)C2)=O)ccc1=O 43428,C1(N(C(C(CCC)OCC)=O)C)CC2CCC(C1)N2C(=O)C(C)c1ccsc1 43429,C1(CNC(C(C)OCCCC)=O)CC2(CC(NC(=O)CS(=O)(=O)N(C)C)C2)C1 43430,c1(NC(C(CC(F)F)NC(CCCN=[N+]=[N-])=O)=O)ccc2c(c1)COC2 43431,N1(C(C2CCN(CC(C)C)CC2)=O)CC(NC(=O)Cc2cnns2)CC12CCC2 43432,Cc1cc(C(=O)NC2CC3CC2N(C(C2(C(F)F)CC(F)(F)C2)=O)C3)cnc1O 43433,c1(OC)cnc2ccccc2c1C(N1CCN(C(C2CNC(=O)N2)=O)C(C)C1)=O 43434,c1(CCC(N2CCCC(NC(C(C)OCOC)=O)C2)=O)cccc(F)c1F 43435,C12(CC(=O)NCCCCNC(c3nccc(N(C)C)c3)=O)CCCCC1C2(F)F 43436,C1(CNC(COc2cccc(C(C)C)c2)=O)Cc2ccccc2CO1 43437,N1(C(C(C=C=C)C)=O)CCCC(C2CCN(C(=O)CCC(=O)OC)CC2)CC1 43438,c1(OC)cccc(C(=O)NC2CC(NC(C3CCC(C(F)(F)F)C3)=O)C(O)C2)c1 43439,Cc1cn(C)nc1C(N1CCCCC1CC(N1CCCC1(C)CO)=O)=O 43440,C1(NC(C2C(C=C)OCC2)=O)CCCN(C(c2ccc(S(N)(=O)=O)o2)=O)CC1F 43441,C(=O)(C(C)(C)CNC(C1CCC1)=O)NC1CC(COC)C1 43442,Cn1cnc2sc(C(=O)NCC(C3CC3)NC(C3CSCCS3)=O)cc12 43443,N1(C(c2c(OC)ccs2)=O)CCN(C)C(CNC(C2CC3(CC(=O)N3)C2)=O)C1 43444,c1(C(N(CC(CN(C(Cc2c(C)cccc2)=O)C)O)C)=O)ccc2c[nH]nc2c1 43445,C1(NC(C=CCCC(C)C)=O)CCCN(C(c2cnn(C3CC3)c2)=O)CC1 43446,c1(CC(=O)NCC(C)NC(=O)CCc2cscn2)nn(C)cc1[N+](=O)[O-] 43447,c1(C(=O)NC2C(NC(C(C)CN3CCCCC3)=O)CCC2)ccc(O)cc1 43448,CC(C)(CN=c1[nH]cnc2ccc(O)cc12)c1nc[nH]n1 43449,N1(C(c2c(C)cn(C)n2)=O)CC(NC(C2COCC(C)O2)=O)C2(CCCC2)C1 43450,Cc1cc2c(C(=O)NC3COCC3NC(c3cc(CO)[nH]n3)=O)nccn2n1 43451,C1(C(N(CCC(C)NC(c2cc(O)nn2C)=O)C)=O)CCC2(CCCCC2)C1 43452,CCCCC(C)CCC(=O)NC1CCN(C(c2ccc(CNC(N)=O)cc2)=O)C1 43453,N1(C(C(C)C(F)F)=O)CC(CNC(C2(c3cccc(C#N)c3)CC2)=O)CC1(C)C 43454,N1(C(C2(C=C)CC2)=O)CC(NC(c2cc(C(F)F)cc(F)c2)=O)CC2(CC2)C1 43455,c1(C(N2CCCC(C(C)NC(c3ccc(Cl)cn3)=O)C2)=O)cc2n(c1)CCOC2 43456,c1(-c2cc(CNC(N3CCCC(CC(=O)OC)C3)=O)[nH]n2)ccc(F)c(C)c1 43457,C(=O)(C1=C(F)CN(C(=O)Cc2csc(C)c2)CC1)N1C(CF)CC(OC)C1 43458,C1(NC(=O)COC(F)(F)F)CCCCCCC1O.CC1CCC2CN1C2=O 43459,n1(C(C)C)cc(C(N2CCC3(CC3NC(=O)C(C)n3cncn3)C2)=O)ccc1=O 43460,c1(C(N(C2CCCC(NC(=O)CC3CC3(Cl)Cl)C2)C)=O)cnc2[nH]ccc2n1 43461,Cc1cnc(S(C)(=O)=O)nc1N1CCC2(C(N3CC(CO)C(O)C3)=O)CC2C1 43462,N1(CCC)CCC(C(=O)NC2CN(C(=O)OC(C)(C)C)C2)C(O)C1 43463,CC1Cn2nc(C(=O)NCCCCCNC(=O)C(F)OC(F)(F)F)cc2C(=O)N1 43464,c1(CC(C)NC(=O)NCC2COCCN2)ccc(F)cc1Cl 43465,C(=O)(C(CCC(C)C)NC(=O)CCC1CCCCC1)Nc1ccc(OC)c(C)c1 43466,c1(N(C)C)ncnc(NC(C2COCCN2C(=O)OC(C)(C)C)=O)n1 43467,c1(N2CC(NC(C(C3CCOCC3)C)=O)C(C)(C)C2)ncc(Br)cc1C#N 43468,C(N=c1[nH]c(=NCCc2nccc(O)n2)c2[nH]ccc2[nH]1)c1c(C#N)cccc1 43469,O=C(CC1(C(=O)O)CCc2ccccc21)N(C1CCCO1)Cc1cc(Br)ccc1F 43470,CC(C)CC(O)CC(=O)NCCn1ccc(C(=O)N(CCCC(C)O)C)c1 43471,C(c1cnc(O)nc1O)=CC(=O)N(CCCNC(c1nc(C)c(C)[nH]1)=O)C(C)C 43472,c1(OC)cc(C(=O)NCC2(O)CN(C(c3cnc(Cl)cc3I)=O)C2)ccc1O 43473,c1(C(=O)OC(C(=O)OC)C2CCOC2)ccccc1CCC#N 43474,C1(c2nnnn2C2CC2)(NCCC(=O)NC2CCCCC2)CCC(=O)NC1 43475,N1(C(CCC2CC(NC(CC(C)c3ccco3)=O)C2)=O)CCOC2CCCCC12 43476,N1(C(CCOCC#C)=O)C2CCC1CN(C(=O)Cc1ccccc1CC)C2 43477,C1(C(=O)Nc2c(C)cc(SC3CC3)cc2)CCc2ccnn2C1 43478,C1(C(N(CC(=O)NC)CC)=O)CC12CCN(C(=O)Cc1ccc(C)nc1)CC2 43479,C1(C(=O)NCC(CN(C(=O)CSCCOC)CC)(C)C)CCCC2CCCN12 43480,C(=O)(CCCC(F)F)NC(c1nc(C(N2CCN(CCCC#C)CC2)=O)cs1)=O 43481,N1(C(CC=CCC)=O)CC2ON=C(CNC(C3CC(S(C)(=O)=O)C3)=O)C2C1 43482,N(C(=NCC)NCC1CCCN(C(C)=O)C1)CC(F)=CC 43483,Cn1ncc2c(C(=O)NC3CN(C(=O)Cn4cc(Cl)cn4)CCC3F)ccnc12 43484,CC1(C)CC(C(N2CCCCC2C2CCCN(C(=O)CS)C2)=O)CO1.CCO 43485,CC12CN(C(=O)C3=COCC3)C(C(=O)NC(c3cscn3)CO)(C1)C2 43486,N1(C(c2c(C)n(C3CC3)cc2)=O)CCOCCC1C(F)(F)F 43487,C1(C(=O)NC(C)(CC(=O)O)c2cccc(F)c2)CCn2nncc2C1 43488,C12(NC(CCCSC)=O)CCN(C(c3cc(O)nn3C)=O)CCC1C2 43489,Cc1cccc(C(O)C(=O)NCCC(C)NC(c2c(C)[nH][nH]c2=N)=O)c1 43490,C(C(S(C)(=O)=O)C1CC1)NC(c1ncccc1F)c1n(CCCOC)nnn1 43491,C1(C)(C(=O)NC2CC(C)N(C(c3ccon3)=O)C2)CCC(C)(C)CC1 43492,CCC(C)CC(C)C(=O)N1CCC(C)(NC(c2cc(=O)c(OC)cn2C)=O)C1 43493,N1(C(C(C)=C(C)C)=O)CCCC1C1(NC(=O)COC2CC=CC2)CC1 43494,N1(C(c2c(OCC#C)nccc2)=O)CCCC(C2CCN(CCO)C2)C1 43495,N1(C(C(C)SC)=O)CCC(NC(=O)COc2ccc(F)cc2F)C(F)(F)CC1 43496,C1(NC(c2ccc(OCC)cc2)=O)CCN(C(c2[nH]c(OC)nc2Cl)=O)CC1C 43497,Cc1ccccc1C(=O)NC1CC(NC(=O)CN2CCCC2CO)C1 43498,N1(C(C2CCC(CNC(c3c(CC)nn(C)c3)=O)C2)=O)CCN(C)C(C(C)C)C1 43499,N1(C(CSc2c(C)n[nH]c2C)=O)CCC(NC(=O)CN2CCCNC2=O)CC1C 43500,N1(c2nnc(C)s2)CCC(CNC(c2ncnc3c(C)csc23)=O)C(F)(F)CC1 43501,N1(C(C(n2cc(CC3(C(F)(F)F)CCC3)nn2)C)=O)CCC2CCCC12CO 43502,C(=O)(C(O)CC(C)C)NCC1CC(N(C(CSCC)=O)C)C1 43503,CC1(CCCO)CCCN1C(=O)Cn1cc(I)nn1 43504,c1(C(N2CC(NC(c3cc(C)no3)=O)C(F)C2)=O)cc(F)c(C)cc1F 43505,C(C(CC(C)C)C(=O)N(C1CC1)Cc1ccoc1)NC(COCC(=O)NC)=O 43506,c1(C(=O)NCC(C(C)C)NC(C(COC)(C)OC)=O)c(C)cc(Cl)cc1[N+](=O)[O-] 43507,C(=O)(C(C)(F)C(F)(F)F)NCC1CCN(C(C=Cc2ccc(C)cc2)=O)C1(C)C 43508,C1(C)(CNC(c2c(C)nn(C)c2)=O)CN(C(c2csc(C)c2N)=O)CCO1 43509,C1(N(C)C)CCOC(C(N2CCN(C(C3COCCO3)=O)CC2)=O)C1 43510,C(=O)(CC(O)CC(C)C)NCCCN(C(=O)C(C)CC(F)F)CC 43511,C12(C(N(C)CC3CCN(C(CC=CCC)=O)C3)=O)CC(CO)(C1)OC2(C)C 43512,CCCCCC(C(=O)N1CCC(C)(NC(c2onc(C)c2C)=O)CC1)C(C)C 43513,C(=O)(C(CCC(=O)OCC)N1CCCC(c2ccn(C)n2)C1)NCCC 43514,c1(C(=O)NCCCC(C)NC(c2cn(C)cn2)=O)nc(Cl)sc1Cl 43515,CC1(C)CCCC(CCNC(C2CCC(CNC(C3CCCC3)=O)O2)=O)O1 43516,CC(C(C)(C)C(=O)NCCC(=O)NC(C)(C)C)NC(c1cc(Cl)ns1)=O 43517,C12(NC(C(CC=CC)CC)=O)CCC(CN(C(c3cnc(OCC)cn3)=O)C1)C2 43518,Cc1cccc(C)c1C(=O)NC1(CNC(=O)C(CO)NC(=O)CCF)CCC1 43519,C1(NC(C2(CC)COC2)=O)CC(NC(=O)C(C)OCC(C)C)CC1O 43520,C1(C(C)NC(C(C)CO)=O)CCN(C(c2cn(-c3ccccc3Cl)nn2)=O)CC1 43521,Cc1nc(C)c(CNC(C2CC2C(C)NC(c2ccc[nH]2)=O)=O)[nH]1 43522,CC1CC(C(c2ccccc2)=O)CCN1C(C1CCCN1C(N)=O)=O 43523,C=C(CNC(=O)NCCC(O)CNC(=O)C)CCOC.C(C)(C)(C)OC(=O)NC 43524,c1(C(=O)NC2CCCC(NC(c3c(C)sc(Cl)n3)=O)C2)cn(C)c2ccccc12 43525,C1(NC(C(C)C2CCCC2)=O)C(C)CCN(C(c2ncc(C(F)(F)F)s2)=O)C1C 43526,C1(C)(CNC(C(C(C)C)O)=O)CCCN(C(c2cccc(Cl)c2F)=O)C1 43527,C(CSC)(CN=c1nc(N(C)Cc2nc(-c3ccccn3)n[nH]2)cc(C)[nH]1)OC 43528,c1(C(=O)NC2C(C)CCN(C(c3cc(Cl)cnn3)=O)C2)ccc2nc(O)oc2c1 43529,C1(CNC(C(CC)n2nccc2C)=O)(OCC)CCCC1C 43530,C1(C(N2CCCC(F)(C(=O)NCc3snc(C)n3)C2)=O)CC(=O)CC12CCC2 43531,N1(C(C)=O)CC(O)CC1C(N1CC(CO)(NC(=O)Cn2nc(C)nc2C)C1)=O 43532,c1(OCCOC)ncccc1C(=O)NCCCNC(=O)CC1CCC(C)(C)C1 43533,N1(C(C(C)OCC=C)=O)CC2CC1C2CNC(=O)C(C)COC 43534,c1(OCCC(N2CCC(C(C)NC(CCC#C)=O)CC2)=O)cc(C)cc(C)c1 43535,C(=O)(CC(C)(C)N(C(=O)CN1CC2CC2C1)C)N(CC(C)C)CC(N)=O 43536,C1(CNC(C(C)SC)=O)CN(C(c2ccc(C(F)(F)F)cc2N)=O)CC1(F)F 43537,C1(CCNC(C(c2cscn2)OCC)=O)CCCN1C(=O)CC1CC(SC)C1 43538,c1(C(=O)NCC2C3N(C(c4c(C)cc[nH]4)=O)C(CC3)C2)cc2ncccc2o1 43539,C1(C(=O)NCC(C2CCCCC2)NC(C(C)n2ccnn2)=O)CCCC(C)(C)O1 43540,C(=O)(C(CO)C(F)(F)F)N(C)CC=CC(=O)NCC1CC(F)C1 43541,N1(C(C=Cc2c(C)nccc2)=O)CC(C)CN(C(=O)C(C)OCC2CC2)CC1C 43542,c1(N(CC(CC)(C)OC)C)nc(=NCC2(C)CC2(F)F)[nH]c2c1CCCC2 43543,C1(C(N2CCN(C(C3CN(C(C(C)(C)O)=O)C3)=O)CC2)=O)CC2(C1)CS(=O)(=O)C2 43544,N1(CCOC)CCN(C(c2ccccc2I)C(=O)NCC2CCOCC2)CC1=O 43545,C1(NC(c2c(C)nc(CCC)o2)=O)COCCN(C(c2ccc(C#N)s2)=O)C1 43546,O=C(N=c1ccn(CCF)[nH]1)C(=O)N1CCC(C(F)(F)CO)C1 43547,C1(CC)CN(C(C2C=CCC2)=O)CCC1NC(c1ccc(=O)n(C)c1)=O 43548,C1(C(=O)NCCOCCCC)CN(C(c2ccc(CC)s2)=O)CC1C1CC1 43549,c1(NC(CC2CN(C(C3(Cl)C(N(C)C)C3)=O)C2)=O)ccc(C2CC2)nn1 43550,C12(C(=O)NCc3cc(C)sc3)CC(C)(CN1C(=O)CC1CC3CCC1O3)C2 43551,C(C(CCC)C(=O)NC1(C)CCCCCC1)NC(C=CCCC)=O 43552,c1(C(N2CCC3CCCC23CNC(C2(CO)COC2)=O)=O)cn2cccnc2n1 43553,C12(NC(CCCC#C)=O)CCCCC1N(C(=O)CCc1ncccc1C)CC2 43554,Cc1cccnc1CC(=O)NC1(CCC(=O)NOCCC2CC2)CCCC1 43555,C1(C(N(CCCNC(=O)CCc2cccc(O)n2)C)=O)CCC2CCCCN12 43556,C(=O)(C(C)(C)CC1CCOC1)NC1C(NC(=O)NC)CCC1 43557,N1(C(CN(C)C)=O)CCC2CN(C(c3cc(C4CCOCC4)[nH]n3)=O)CCC12 43558,N1(C(C2(CC#C)CCCO2)=O)CCC(NC(=O)C(CCO)N(C)C)CC1 43559,CC(C)(CC(F)F)C(=O)N1C2CCC1CC(NC(c1ccc3ccnn3c1)=O)C2 43560,CCC(CCCC(=O)NCC1(CF)CCC1)NC(c1cc(OC)n(C)n1)=O 43561,c1(CC(=O)NC2C(CNC(c3c(OC)scc3)=O)CC2)nn(C)c2ccccc12 43562,C1(NC(C=C(C)C)=O)CCN(C(c2ccc(Br)cc2C)=O)C2CC12 43563,N1(C(=O)NCC)CCC(C)(OC)CC1.N12CC(CO)(CC1C)CNC(=O)C2=O 43564,N1(C(CS(=O)(=O)NCC)=O)CCC(NC(c2ccn3ccsc23)=O)C(C(C)C)C1 43565,O=C1CCC(CNC(c2ccc(CNC(=O)CC3CCCO3)s2)=O)O1 43566,C1(NC(=O)Cn2ccnc2)CN(C(c2cccc(C(F)(F)F)c2F)=O)CC1(F)F 43567,N1(C(C2(CC)CCC2)=O)CC(C)(CNC(=O)CNC(C2CCCC2)=O)CC1(C)C 43568,c1(C(=O)NCCCCCCNC(C2C(CCC)C2)=O)c(Cl)cnc(OC)c1Cl 43569,C1(C(N(C2CCCOC2)CC)=O)CC12CCN(C(C1CC3CC(=O)C1C3)=O)CC2 43570,N1(C(C(C)=C2CC2)=O)CC(C)CN(C(c2nc[nH]c3nccc2-3)=O)C(C)C1 43571,c1(Nc2ccc(C(=O)OC)nc2I)c([N+](=O)[O-])cc(C(F)(F)F)cc1[N+](=O)[O-] 43572,n1(C(C)C)cc(C(=O)NC23CC(NC(=O)C(F)F)(C2)C3)cn1 43573,C(CCCC(F)(F)F)N(C=O)CCN1CC2CCC1C2 43574,C1(CC)(CC)CCN1C(=O)OC(C)(C)C 43575,CCCC(O)C(=O)N1CCC(N(C(=O)CC(C)C2CC2)CCC)C1 43576,C(CN=c1[nH]c2ccc(Br)cc2s1)N(C(=O)CCC1CC1CO)CCC1CC1 43577,CC(C)(C)CCCNC(=O)NCCN1CCCC(N(C)C)C1 43578,C1(C(C(=O)OC)NC(=O)C=CCN)CCS(=O)(=O)C1 43579,C(CCC(=O)N1CCN(CCO)C(C)C1)(C(C)C)NC(c1c(C)coc1)=O 43580,C12(C(N(C)CC3COCCN3C(=O)CCCn3cccc3)=O)CCC(C1)C2(C)C 43581,C(=O)(CC(C)(C)CNC(=O)CC1CCCCC1O)N(C)CC 43582,Cc1ccccc1CC(=O)N(C1CN(C(c2cnn(CCO)c2)=O)CC1F)C 43583,N1(C(C=CC=CC)=O)CC(CNC(=O)Cc2cc(C(F)(F)F)co2)OC2CCCC12 43584,C1(C)(CNC(C2C=CC(NC(C(C)n3cccc3)=O)C2)=O)NC(=O)NC1=O 43585,c1(C(N(C2CN(C(C(CCCC)CC)=O)CC2O)C)=O)ccnc2c1CC(=O)N2 43586,N1(C(C=CC(CC)C)=O)CCC(NC(c2cnc(N(C)C)s2)=O)C(O)C1 43587,CC(C)C(O)CC(=O)NCC1CC(F)CN1C(=O)C=Cc1cc[nH]c1 43588,C1(C(=O)NCc2cnco2)(NC(=O)Cc2ccsc2)CCCCC1 43589,CC(C(=O)NC1CN(C(c2ncccc2N)=O)CCC1c1ccccc1)C(C)(C)C 43590,C(=O)(C(F)C(F)(F)F)N(CCC)CCNC(C1CCC1C(C)(C)C)=O 43591,C(=O)(C1CCc2cccnc21)NCC1CN(C(C2(OC(C)=O)CC2)=O)CC12CC2 43592,N1(C(CCSCCCC)=O)CC(CNC(c2cc(OC)cnn2)=O)CC1C 43593,c1(OCC(=O)N(CC(CNC(C(C)O)=O)O)C)cccc(Cl)c1 43594,c1(NC(c2cccc(NC(c3cnc(Cl)nc3)=O)c2)=O)cc(Br)cnc1O 43595,C1(C(N2C(C(C)(C)NC(c3[nH]cc(CC)c3)=O)CCC2)=O)CCCN(C)C1 43596,Cn1c(C(N2CCC(C)(CNC(=O)C(O)C(F)F)CC2)=O)c(Cl)c2ccccc12 43597,CCC(CC)C(=O)N1C(CNC(c2cc(CC(C)C)nn2C)=O)CC2CC12 43598,c1(C(=O)NCCC(=C)CNC(=O)CC2CN(C(=O)OCC)C2)cc(C)ccc1Cl 43599,Nc1cc2ccccc2cc1C(N1CCC2CN(C(C34CCCC3C4)=O)CC12)=O 43600,C1(NC(CC(C=C)(C)O)=O)C2CC(CN(C(c3coc(Br)c3)=O)C2)C1CO 43601,C1(C(N(C2CCN(C(=O)CCCc3cnn[nH]3)C2)CC)=O)CCN(C2COC2)C1 43602,C(=O)(C1=NNC(=O)C1)NCC(C)(C)NC(C1CN(C2CCOC2)C1)=O 43603,C1(C(=O)NCC(CNC(CCCOCC)=O)(C)C)CCCC12OCCO2 43604,N1(C(c2c(SC)n(C)nc2)=O)CC(C)CN(C(c2ccc(Cl)cc2Cl)=O)C(C)C1 43605,c1(CNC2CC(C(=O)NCCC(F)(F)F)C2)ccc(F)c(F)c1Br 43606,C1(C(N(CC(C)(C)CO)C)=O)C(C2CC2)CCN1C(c1ncccc1Cl)=O 43607,Cc1nc(C)c(CNN(C(C2N(C(CSc3cccc(F)n3)=O)CCC2)=O)C)[nH]1 43608,C1(NC(C(CC=CC)CC)=O)CCCCCN(C(c2ncsc2CC)=O)C1 43609,Cc1nn(CC(=O)NCCCN(C)C(C2CCC(C3CC3)C2)=O)c(=O)n1C 43610,c1(CN(C(=O)C(F)n2ccnc2)CCNC(CSC)=O)ncnn1C 43611,C1(OC)(CNC(=O)CC2(Sc3ccnn3C)CC2)CN(C(CCCC(C)C)=O)C1 43612,c1(N(C)CCn2ccnc2)[nH]c(=NCCn2ncnn2)nc2scnc12 43613,Cc1c(C(=O)NC(C)C(C)NC(=O)Cc2ccc(Br)cn2)noc1C1CC1 43614,c1cc(NCC2CCC2C2CC2)cc(-n2cnnn2)c1 43615,c1(NC(CC)C)cc(N(C)CCn2cccn2)nc(COC)n1 43616,Cc1oc(CO)cc1C(N1CCOCC1CC(=O)NCC1CCC(C)C1)=O 43617,c1(C(C(=O)N(CCOCCCNC(CCSCC(C)C)=O)C)O)ccnn1C 43618,Cc1cc(C(=O)NC(C)(C(=O)NCCc2cc(C)ns2)C2CCC2)ccc1C#N 43619,c1(C(=O)NCC23N(C(c4cc(C)c(C)o4)=O)CC(C2)C3)cccc(C=C(F)F)c1 43620,C1(C(N2CC(NC(C(C)Cn3cccn3)=O)C2)=O)C2C3CCC(C3)C12 43621,C1(CNC(C(C=C)(C)CC)=O)CN(C(C2OCCO2)=O)CCC1(F)F 43622,c1(C(=O)NCC(CN(C)C)NC(=O)OC(C)(C)C)ccc(=NC(=O)OC)[nH]n1 43623,C1(NC(=O)Cc2ccc(O)cn2)CN(C(=O)C2=CCCSC2)C2(CCCOC2)C1 43624,N1(CC#C)CCN(C(C2CCN(C(C3CCCCO3)=O)C23CC3)=O)CC1=O 43625,c1(CCNC2CC(C)N(c3ccccc3)C2)cc(O)nc(O)n1 43626,Cc1ccnc(C(N2CCC(n3cc(Cc4ncc(F)cn4)nn3)C2)C)n1 43627,c1(SCC)ncc(CN2CCC(C)(N3CCCC3)C2)cn1 43628,CC(C(=O)N1CCN(CCNC(C2CCCN(C(=O)C(N)=O)C2)=O)CC1)C(F)F 43629,N1(C(C=C(C)C(F)F)=O)CC(NC(c2ccncc2C(F)F)=O)CC(O)C1 43630,C1(C)(C(=O)NCCc2c(CNC(C(C)n3ccnn3)=O)nco2)CCC12CCC2 43631,N1(C(c2cc(CC#C)on2)=O)CCC(C(F)CNC(C2CC2C#C)=O)CC1 43632,c1(NC)cnc(C(N2CC(CNC(c3n[nH]cc3Br)=O)C(C(F)(F)F)C2)=O)cn1 43633,Cn1c(C(=O)N(CCCN2CCc3ccccc32)C(C)(C)C)cc2ccsc12 43634,C=CC(C)(C)CCCNC(C1CC(NC(c2cc(C)c[nH]2)=O)C12CCC2)=O 43635,CCCC(C)CCCC(=O)N1CC(O)(C(C)NC(c2cnnn2C)=O)C1 43636,c1(C(C)=O)cc(C(N2CC(CC(C)NC(c3csc(CO)n3)=O)C2)=O)no1 43637,CC1(CC(N2CC(C#N)C2)=O)CCN(C(C2CCNC2=O)=O)C1 43638,Cc1ccccc1C1(C(=O)NC2C3CC2N(C(=O)COCCN(C)C)C3)CC1 43639,C12(C(=O)OC)CCC(C(N3CCC(C)C(NC(=O)C(C)SC)C3C)=O)(CC1)CC2 43640,N1(C(c2cnc(Cl)s2)=O)CCC2CCCC12CNC(C1(C2CC2)CCOCC1)=O 43641,C1(C(N(CC(CNC(c2c(C)nc(O)[nH]2)=O)(C)C)C)=O)CC2CCCCC2O1 43642,C1(C(C)C)C(=O)NCCN1C(C1C2CCC(C2)N1C(c1cc(C#N)cs1)=O)=O 43643,n1(CC(N)=O)cc(C(=O)NCC(C2CC2)NC(c2n[nH]cc2Br)=O)nn1 43644,N1(C(C=CCCC(C)C)=O)CCCC(NC(c2ccc(CC(C)(C)C)cc2)=O)C1 43645,c1(C(=O)NC(C)C(C)(C)NC(C2(C3CCCO3)CC2)=O)cc2sc(Cl)cc2s1 43646,N1(CCC)CC(C(=O)NC2(CNC(=O)CCCC3CCCC3)CCCC2)CC1=O 43647,N1(CCNC(C(C)SC)=O)CCN(C(=O)CNc2nccc(OC)n2)CC1 43648,C1(C(=O)NCCc2nc(CC)[nH]n2)CCN(C(=O)c2cccnn2)O1 43649,CN1CC(C)(C)CC1C(N1CC(NC(=O)C2=C(Cl)CC2)C(O)C1)=O 43650,C1(C(=O)NCC(CC(=O)NC(C)C(C)C)OC)CC2(CCC2O)C1 43651,c1(CC)nc(CC(=O)NCC(C2CCOC2)NC(=O)COCc2cccs2)cs1 43652,N1(C(CC=C)=O)CC(NC(C2(C(=O)OCC)CCCO2)=O)C(c2cnn(C)c2)C1 43653,C1(NC(c2ccc(C(F)(F)F)nc2)=O)CCOCC1NCC=CC=C(Cl)Cl 43654,N1(C(Cc2c(OC)cccc2)=O)C(C)C2CC1C2NC(=O)CCn1cc(C)cn1 43655,CS(=O)(=O)CCC(=O)NCC12CCC(CC1)N2C(c1cncc(OC2CC2)c1)=O 43656,C1(CNC(c2c(Cl)nsc2Cl)=O)CC(F)(F)CN1C(C1CCCC12CC2)=O 43657,c1(C(=O)NC2CN(C(C=CSC)=O)CC2C(F)F)cccc2[nH]ccc12 43658,N1(C(C(C)c2ccsc2)=O)CCOC2(CCN(C(c3ccc(F)o3)=O)CC2)C1 43659,CCCC(C)(O)CC(=O)N1CCCCC(CNC(=O)CCNC(C2CCC2)=O)C1 43660,c1(OC)cccc(C(=O)NC2CC(CCNC(C3CCC(=O)NC3)=O)C2)n1 43661,Cc1nc(CC(=O)N(C)CCN(C(=O)C2=CCCC2)C)c(Cl)s1 43662,c1(OC)ccc(Cl)c(F)c1C(=O)NC(C1CCOC1)CNC(c1occc1C)=O 43663,c1(OC)cc(C(N2CC(NC(c3oc(Br)nc3C)=O)C2)=O)cc(N)c1O 43664,c1(CC)nc(C(=O)N(C)CC2(NC(=O)CC3(CO)CC3)CC2)cs1 43665,Cc1occc1S(C)(=O)=NC(=O)CC1(C)CC1 43666,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC1CCN(C(C(C)(CO)OC)=O)C1 43667,C(=O)(CC(C(F)(F)F)NC(c1ccc2ccoc2c1)=O)NC(CCC)C1CCC1 43668,N1(C(COC2(C)CCC2)=O)CCC2(CCN(C(C3CCCO3)=O)C2)C1 43669,C1(CNC(c2cncc(C)c2)=O)CCC(C)N(C(=O)CCc2cncnc2O)C1 43670,C12CCCCC1N(CCN(C)CCO)C(=O)C2.C(=O)(CC1CC1)NC1CSC1 43671,N1(C(CC2CC(=C)C2)=O)CCC(N2CC(O)C2)C1(C)C.N12CCC(C1)C2=O 43672,CN1CCC(C(=O)NCC2CCC(NC(=O)CN3CCC(O)CC3)C2)CC1 43673,Cc1cc2sc(C(N3CC(F)(CNC(=O)C(C)n4ccnc4)C3)=O)cc2s1 43674,N1(C(C2(C#C)CN(C(=O)C(O)CN3CCCC3)C2)=O)CCC(C2CCC2)C1 43675,c1(C(N(CC(C)NC(c2cnc(Cl)c(N)c2)=O)C)=O)cnc2ncc(Cl)cn12 43676,c1(CC)cccc(C(=O)N(CC(C)CNC(=O)C=CC2CCCN2C)C)c1F 43677,c1(C(=O)NCCCCCN(C(CC2(CC)CC2)=O)C)c(C(C)C)cccc1C 43678,c1(N)cccc(=O)n1C.C1(C(=O)Nc2cn(N3C(=O)C3)nc2)CCCC1c1ccccc1.CC 43679,CS(=O)(=O)C(CNC(=O)CC1CCCOCC1)CNC(C1CC(F)(F)CS1)=O 43680,C1(NC(C2CCCN(CCC)C2)=O)C2CC1CN(C(=O)CCN1CCCC1=O)C2 43681,C(=O)(CC(C(C)(C)C)NC(=O)Cc1cncs1)NCC(CN(C)C)O 43682,Cc1cncc(C(=O)NCC2CCN(C(=O)Cn3ccc(=N)[nH]3)C2)c1 43683,C1(C(=O)OC)CCc2cc(OC)ccc2N1C(C1(C)CC1(F)Cl)=O 43684,c1(C(=O)NCC2CCCN(C(=O)C=C3CCSCC3)C2)c(F)cccc1[N+](=O)[O-] 43685,N1(C(C(C)C)=O)CCN(C(=O)CSc2nc(-c3ccccc3)no2)C(CF)C1 43686,C(=O)(C(CNC(c1n[nH]c2c1COC2)=O)CC(C)C)Nc1c(C)ncnc1 43687,C(=O)(C(C)(C)C(C)NC(c1c[nH]c(C)cc1=O)=O)Nc1c(OC)nsc1 43688,c1(C(N(CCNC(C2(CC=C)CC2)=O)C)=O)cccc2ncnc(O)c12 43689,N1(C(C2CCCN(C(CCCCC=CC)=O)C2C)=O)CC(C)CCCC1C 43690,C1(NC(CCc2onc(C)n2)=O)CCN(C(=O)CCc2scnc2C)CC1(C)C 43691,CS(C)(=O)=NC(=O)C(=O)NC1CN(C(C2CCCN2C(C2CCCC2)=O)=O)C1 43692,c1(C(=O)NCC(C)N(C(C(C)=C2CC2)=O)C)ccc(-c2cc[nH]n2)cc1 43693,N1(c2cc(N3CCC(CN(CC)CC)C3)nc(C)n2)C2CCC1CC(CC)C2 43694,CC1CC2(CCN(C(=O)CCN3CCCC3=O)CC2)CN1C(C1CCC1(C)C)=O 43695,c1(OC)ccc(O)cc1C(=O)NCC1(NC(c2nnn(C)c2C)=O)CCOC1 43696,N1(C(COC(C)=O)=O)CCCC12CCN(C(=O)Cn1cc3ccccc3n1)C2 43697,C1(CC)CN(C(=O)C(C)C2(O)CCC2)CC1C(=O)NCc1nccn1C1CC1 43698,C1(C)(C(N(CCC(=O)NC2C(C)CCCC2)CCCO)=O)C(C)(C)C1(C)C 43699,CC(C)C(F)C(=O)NC1CCCC(NC(C2(c3ccccc3)CC(F)(F)C2)=O)C1 43700,C1(C(=O)NCc2cccc(OC(F)F)n2)CCc2nc[nH]c2C1 43701,C=C(C)C(C)(O)C(=O)NC(C)CN(C(c1cc(Br)ccn1)=O)CC 43702,C12(C(=O)OC(C(=O)NCC)C)CCC(CC1)C2(C)C 43703,C1(CCOC)OCCC1Nc1ncc(I)s1 43704,c1(C(=O)NCC2CCN(C(C(CCC)O)=O)C2(C)C)ccc2cc(Cl)ccc2n1 43705,c1(C(=O)NCC(C2CCCN(C(C3CS(=O)(=O)C3)=O)C2)(C)O)cnc2sccn12 43706,c1(CC)cnc(Cl)[nH]c1=NC(CNC(c1ccc(C)c(Cl)c1)=O)c1ccccc1 43707,C1(CNC(C(CC)NC(N)=O)=O)CCCN(C(C2(CO)CCC2)=O)CC1 43708,N1(C(c2c(N)ccc(F)c2)=O)CCN(C(c2ccc3[nH]ccc3c2)=O)CC(O)C1 43709,CC1C(C(=O)N(C(C)(C)CC(N2CC3C=CC2CC3)=O)C)=NOC1C 43710,c1(C(N(C2CCN(C(c3cnnc(O)c3)=O)C2)CC)=O)cnn2ccn(C)c12 43711,C#CCCC(O)CCNC(=O)CC1CCCN(C(=O)C(CC)(CC)OC)C1 43712,N1(C(c2nccc(CC)c2)=O)CC2CCC2(NC(c2cnc(C3CC3)s2)=O)C1 43713,N1(C(C2CC(OC)CN2C(=O)Cc2cccc(O)c2)=O)CC(F)(F)CC1CO 43714,C1(CC(=O)N(CCCCN(C(c2cc(C)sc2)=O)C)C)CCOC(C(C)C)C1 43715,c1(CCNC(c2occc2C(=O)O)=O)cccc(F)n1 43716,C(=O)(C(O)CC(C)C)N1CC(NC(C(=C(C)C2CC2)F)=O)C(C)C1 43717,CCCC(CC)C(=O)N1CCN(C(=O)CCCOc2ccc(F)c(F)c2)C(C)C1 43718,C(N=c1[nH]c2c(c(=NC3CCc4cccc(Cl)c43)[nH]1)SCC2)c1ccc(O)nc1 43719,C(CC(CC)C(=O)N1CC(NC(=O)C=Cc2cncc(F)c2)C2(CC2)C1)=CC 43720,Cc1ncc(C(N2CC(C)(NC(=O)CCC3CC(C)C3)C2)=O)cc1C#N 43721,c1(C(N2CCN(C(C3C(C(N)=O)C3)=O)CC2)=O)ccc2c(c1)COCC2 43722,c1(CC)csc(CC(=O)NC2(CCNC(c3cc(C(C)(C)C)on3)=O)CC2)n1 43723,c1(CNCC(c2ccccc2)F)cc(Cl)cc(Br)c1 43724,c1(CC)ccc(C(F)(F)F)nc1SCC(C)(C)NC(=O)NC1(C(F)(F)F)CCCC1 43725,C1(NC(c2cc(OC)ncc2)=O)CCN(c2ccnc(C(F)(F)F)n2)CC1C 43726,C(C(C)C)(C(O)C(=O)NCC1CN(C(=O)C(C)(C)OC(C)C)CC(C)(C)O1)OC 43727,C1(CC(=O)NCCCCCN(C(CC(C)C)=O)C(C)C)CC(C)(C)CO1 43728,C(C(C(C)C)NC(c1cn(CCNC(c2ccc(Cl)s2)=O)nn1)=O)OC 43729,N1(C(CCC(=O)NC)=O)CCC2(CC1)CC2(C)C(=O)NC(C)C(C)(C)C 43730,Cc1cc(C(=O)NCC2CC(NC(=O)CC3CCC(C)CC3)C2)cc(N)c1 43731,C1(NC(=O)CCc2cnc[nH]2)CC12CCN(C(=O)C=CC=C(Cl)Cl)C2 43732,C1(CC)CCN(C(c2c[nH]ccc2=O)=O)C(C(N2CC=CC2CF)=O)C1 43733,N1(C(C(=O)Nc2cccc(C)c2C)=O)CC(C2CN(C(=O)CC3CC3(Cl)Cl)C2)C1 43734,c1(CC)c(C(=O)Nc2cccc(-n3cc(CCC(C)O)nn3)c2)cnn1C 43735,CC1CCN(C(c2ccc(Cl)c(N)c2)=O)CC1NC(c1c(Cl)nsc1Cl)=O 43736,C1(C(N(C2CN(C(=O)CC3CCCCCC3)C2)C)=O)CN(S(N)(=O)=O)C1 43737,C1(N(C)C(C2COCCC2NC(C2(F)CCCC2)=O)=O)CCCCC1(C)C 43738,c1(OCC(N2CC(CCN(C(C=CC(C)C)=O)C)C2)=O)ccccc1 43739,N1(C(C2N(C(C(COCC)(C)C)=O)CC(=O)C2)=O)CC(C)CCC1CC 43740,C1(CNC(C(C)SC(C)C)=O)CCC(F)(CNC(C2CN(C)C2)=O)C1 43741,c1(C(=O)NC(C(C)N(C)CCNC(c2cccnc2)=O)=O)cccc(N(C)C)n1 43742,N1(C(C(C)Cc2ccccc2)=O)CCCN(C(C23CC(C)(C2)C3)=O)CC1CO 43743,C1(C)(C(=O)NC(C)CCCCO)CCN(C(=O)Cn2ncnn2)CC1 43744,C1(CNC(CCC(=C)C)=O)CC2COCC2N1C(C1CC2CCCC12)=O 43745,c1(C(=O)NCC(CNC(c2c[nH]c(=NC)o2)=O)F)ccc2nccnc2c1 43746,c1(CC(=O)NC(CNC(C2N(CC)CCCC2)=O)(C)C)ccc(OC)c(Cl)c1 43747,C1(CCC)CN(C(c2cc(C)[nH]n2)=O)CC1C(=O)NCCn1cncn1 43748,c1(C(N(CCN(C)CC2(COC)C=CCC2)C)=O)nccnc1SC 43749,C#Cc1ccc(CCC(=O)NCC(C)NC(=O)CN2CCOCC2)cc1 43750,N1(C(CC)=O)CC(C(=O)NC(CCC)C(=O)NC)C2(CCC2)C1 43751,c1(C(c2n(CC=C)nnn2)NC2CCCCN2C)ccc(C(=O)NC)cc1 43752,C1(C2CCCN(C(=O)C(C#N)C(C)(C)C)C2)(NC(COC)=O)CC1 43753,C1(CC(=O)NC2(CC(N)=O)CCC2)CCCN1C(=O)CC1CCC1 43754,N1(C(C(CCC)N(C)C)=O)CC2(CNC(=O)CCc3ccon3)CCC1C2 43755,Cc1ccnc(C)c1NC(C1CC2CC2N1Cc1cc(Br)cnc1F)=O 43756,c1(C(C(=O)NCCC2N(C(C(F)=C(C)C)=O)CCSC2)C)c(C)nn(C)c1C 43757,O=C1CCC(C(N2CCC(CNC(=O)C(O)CCc3ccccc3)C2)=O)CCO1 43758,c1(C(=O)NC(CNC(CCN(CCC)C)=O)CC)cc[nH]c1COC 43759,c1(CNC2CCC(NC(=O)CC3CCCCO3)C2)cc(F)cc([N+](=O)[O-])c1 43760,C#Cc1cncc(C(=O)NC2CCC2NC(=O)Cc2ccc(F)c(Cl)c2)c1 43761,c1(N2CC(C)CC(OCC)C2)ccc(S(=O)(=O)N2CCSC(C)(C)C2)cn1 43762,n1(CC(=O)NC(C)CCNC(=O)C(C)(C)CF)ccc2cc(F)ccc12 43763,C(c1ccncc1C)=CC(=O)N(C(CNC(C(CCOC)OC)=O)C)C 43764,c1(C(=O)NC2C(CNC(C(n3cc(C)nc3)(C)C)=O)CC2)cc2nc[nH]c2cn1 43765,Cc1ccc(C(=O)NCC2CC(F)(CNC(C3(C(C)(C)C)CCCC3)=O)C2)nc1 43766,c1(C(C)=O)cc(Cl)c(NC(C2CC3CC3N2Cc2ncc(Cl)s2)=O)c(Cl)c1 43767,N1(C(CC2C(C)(C)CC2)=O)CC2(CCOCC2)CC1CNC(c1csc(S)n1)=O 43768,c1(C(=O)NCC(CN(C(C2=C(C)OCC2)=O)C)(C)C)cc(=O)c2ccccc2o1 43769,C1(C(=O)NC2CC(C(N(CC#C)CC3CCCO3)=O)C2)CC1C1(C)COC1 43770,c1(CC)cnccc1C(N1CCCC1C(=O)OC)C(=O)NC(C)CC 43771,C(=O)(CCCCC(F)F)NC1(C)CCCN(C(c2cccc(CCC)c2)=O)C1 43772,c1(CC(=O)N(CC(O)CN(C)C(C2CC2C(C)(F)F)=O)C)ccnn1C 43773,C(=O)(CCN=c1[nH]ccs1)NCC(CN(C(C1COCCC1(F)F)=O)CC)(C)C 43774,c1(C(=O)NCC(CNC(=O)CC2CCCC2O)CO)nccc2ccncc12 43775,N1(C(CNC(CC)=O)=O)CCN2CCN(C(=O)CC3CCCC(=O)N3)CC2C1 43776,C=CCC(C)(C(=O)N1CCC(N(C(c2cc(C)ncc2C)=O)CC)C1)N(C)C 43777,C(=O)(C(CC)N(C)C(c1ocnc1C)=O)NC1CN(C(CC)=O)C1 43778,C(CC(C)(C)C(=O)NCC1COCCN1C(=O)C=CC(=O)NC1CC1)OC 43779,C1(NC(C(CC=CCC)C)=O)CC2CCC(C1F)N2C(=O)C(C)(C)F 43780,C(=O)(C(C)S(C)(=O)=O)N1CCC(N(CC#C)C(c2cccs2)=O)C1 43781,C1(CCNC(C(C)n2cnnn2)=O)CCCN(C(c2cnoc2)=O)CC1 43782,c1(C(=O)NC2C(NC(CCOC(C)C)=O)CC2)cnc(Cl)c(N)c1 43783,C1(NC(CCCCC=CC)=O)CN(C(C2NC(=O)OC2(C)C)=O)CC2(CC2)C1 43784,C1(C(=O)NCCCNC(CC2CCC(C)C2)=O)CC=CC(O)C1 43785,N1(C(CCC2CCC(=O)C2)=O)CC2(CCC(NC(=O)C(C3CC3)C3CC3)CC2)C1 43786,C(CCC(O)C(=O)NCCCCn1ccnc1)NC(=O)CN1CC2CC2C1 43787,c1(C(=O)NCCCC(C)NC(C2CC(=C)C2)=O)cc2ccc(F)c(F)c2o1 43788,c1(C(C)C)nc(CC(=O)NC(C2CCCN2C(C2CC(F)C2)=O)C)cs1 43789,C1(CC)CCN(C(=O)C(C)=CC(C)(C)C)C1C(N1CC(OC(=O)N(C)C)C1)=O 43790,c1(-n2c(C(=O)NCC(C)NC(C3(COC)CCOC3)=O)cnn2)ccccc1F 43791,c1(OC)ccc(CNC2CCC(C(=O)O)C2)c(O)c1 43792,CON(Cc1ccco1)C(=O)C(F)CC(C)(C)NC(=O)CC1CC(SC)C1 43793,N1(C(c2c(CC)cccn2)=O)CC(CC(=O)NCCN(CC(F)F)C)CC1(C)C 43794,Cc1cc2nc(C(=O)NC3CC(C)N(C(=O)CCCCC4CC4)C3)cn2cc1C 43795,O=C(C(F)C(F)(F)F)NCC1CCCCC1C(=O)NCC1CC2CCC1O2 43796,C1(NC(c2ccc(CNC(C3OCC(C)C3)=O)cc2)=O)CCC(=O)NC1C 43797,c1(-c2cn(CC3C(NC(c4ccc(SC)s4)=O)CCC3)nn2)c(C)cccc1C 43798,N1(C(C2CCCCC2O)=O)CC2CCCN(C(C3CC34CCC4)=O)C2C1 43799,C#CCCCC(C)C(=O)NC(c1nccs1)CC 43800,C1(NC(c2n(CCC)nc(C)c2)=O)CC2CN(C(=O)CCC(C)(C)F)CC2C1 43801,S(=O)(=O)(c1cc(C)c(Br)cc1F)NC(C(CCC)OCC)=O 43802,C1(NC(C2CCN(C(CC(C)(F)F)=O)CC2)=O)CCCCCC1O 43803,N1(CC(=O)NC(CC)CO)CCC(N2CCC(C)(O)C2)CC1 43804,c1(C(=O)NC23CC(CNC(CCC(C)SC)=O)(OCC2)C3)ccn2cnnc2c1 43805,N(C(=NCCC(=O)NC1CC2(CC(OC)C2)C1)NCc1ccccc1)CC(CC)C 43806,C(=O)(CCCCC(C)(C)OC)NC(C)C(C)NC(c1c(OC)c(F)ncc1)=O 43807,C(c1cc(F)cc(F)c1)=CC(=O)NCC(C(C)C)NC(C(C1CC1)SC)=O 43808,N1(C(c2ccn(CCC)n2)=O)CCC2(CCN(C(c3cc(N)ccc3C)=O)C2)C1 43809,c1(-n2cc(CCN(C)CCN3CCNCC3)nn2)c(C(F)(F)F)nc2ncccn12 43810,c1(NC2(CNC(CSc3c(C)cccc3)=O)CCCC2)c(Cl)cccc1[N+](=O)[O-] 43811,N1(C(CCC2CC(NC(c3c(C)n(C)nn3)=O)C2)=O)CCC(N(C)C)C(C)C1 43812,C(=O)(C(F)(F)CN)NCC(Cc1ccccc1)OCC 43813,c1(C(=O)NCC(C)(C)NC(C(CC)C(C)O)=O)ccc2c(O)nc(=O)n(C)c2n1 43814,c1(NC(C(C2CN(C(CC3CC(=C)C3)=O)C2)O)=O)ccc(F)cc1C 43815,c1(OC(C)C(=O)NCC(F)CNC(c2csnn2)=O)ccc2c(c1)CCC2 43816,C1(CNC(C(C=CCCC)O)=O)(NC(c2cc(O)cs2)=O)CCCCC1C 43817,N1(C(=O)Nc2c(C(=O)OC)cnn2C)CC(NC(c2ccccc2)=O)C2(CC2)C1 43818,N1(C(C2(SC)CC2)=O)CC(NC(=O)C(O)CC2CCCCC2)C2(CC2)C1 43819,C(=O)(CC(CNC(=O)CC1(C)OCCO1)C1CCC1)N(CC(C)C)C 43820,C=CCC(CNC(=O)C(=O)C1CC1)CC(C)C(C)(C)C 43821,Cc1ccc(O)cc1C(N1CCN(C(=O)Cc2ccon2)C(C)C1)=O 43822,CC1(C)CCN(C(=O)C2CC2)CC1CNC(C1CC(NC(c2ccsc2)=O)C1)=O 43823,C=CCCCCC(=O)N1CCC(CF)(NC(c2cnccc2Cl)=O)C1 43824,C1(CNC(C(N2C(CC)CCC2)=O)=O)CSCCN1C(=O)CSCCN(C)C 43825,c1(C(N2CC(CNC(CC=CCC)=O)C(F)(F)C2)=O)cccc2nc(Cl)cn12 43826,S(=O)(=O)(c1cccnc1NCCc1cscn1)NCc1ccc(OC(C)C)nc1 43827,N1(C(c2cnc(CC)o2)=O)C(CC(=O)NC2C=CCCC2)C2CCCC12 43828,c1(CC(N2CCN(C(CN(C(C)C)C)=O)CC2)=O)cccc([N+](=O)[O-])c1 43829,c1(C(=O)NCC2CC(F)(CNC(CS(=O)(=O)NC)=O)C2)ccc2c(c1)ncn2C 43830,c1(C(CNC(=O)NCc2c(C)nc(CC)o2)N)cccc(Br)c1F 43831,c1(OC)nc(C(=O)NCC(N2CCN(C(c3cc[nH]c3C)=O)CC2)C)ncc1F 43832,C1(O)(C(CNC(CC=C=C)=O)C)CCN(C(=O)CC2(C)CCOCC2)C1 43833,C1(O)(C(=O)NCCN(C(=O)C(c2cccc(C(F)(F)F)c2)(C)C)CC)CC(F)(F)C1 43834,N1(C(C(CCN(C)C)NC(c2cc[n+]([O-])cc2)=O)=O)CCCCCCCCC1 43835,N#Cc1ccc(F)c(C(N2CCC3CCC23CNC(c2csnc2Cl)=O)=O)c1 43836,CC1CCN(CCCCn2c(N3CCSCC3c3cccs3)nnc2C)CC1 43837,c1(C(=O)NC2(CNC(=O)CC3(C(F)F)CC3)CCOC2)cc(O)cc(Cl)c1 43838,c1(CC(=O)NC2CC(C)(NC(c3ccsc3Br)=O)C2)nc2ncccn2n1 43839,C1(CNC(COC(CC)(C)C)=O)CCCC1NC(=O)C=Cc1cncs1 43840,CC1CN(C(c2cncn(C)c2=O)=O)CCC1NC(c1cc(C2CCC2)[nH]n1)=O 43841,c1(OCC)nccc(C)c1NC(=O)CCC(C)NC(C1C=CCCC1)=O 43842,c1(C(=O)NC2C(F)CCN(C(C3(C)CCOCC3)=O)C2)cccc2ccsc12 43843,C(CC(C)C(=O)N(C(C)CNC(C1(C)SCCCS1)=O)C)=CC 43844,C1(NC(C2CC(CCC)C2)=O)CCC2(CC1)CCN(C(c1cccnc1O)=O)C2 43845,c1(C(=O)NCC2(COC)CN(C(C3CC(C)CO3)=O)C2)ccc(C)cc1C 43846,C(=O)(CC(C)C(F)F)N1CCCC(NC(c2nc(COC)sc2)=O)C1 43847,c1(CC(C)C)cc(C(=O)NC2CN(C(c3ccc(C4CC4)o3)=O)C3CC23)n(C)n1 43848,c1(C(N2C(C)(C(=O)NCc3ccc(O)c(O)c3)CCC2)=O)ccc2nn[nH]c2c1 43849,Cc1c(C(=O)OCCC2CCN(C)C2=O)sc2nc(C(F)(F)F)ccc12 43850,N1(C(CC=C(C)C)=O)CC2CC2(CNC(=O)CCSC(F)(F)F)C1 43851,c1(N2CCC(CN(C(CC)C(=O)NC)C(C)=O)C2)nc(CC)nc2ccccc12 43852,c1(CC(=O)NC2CCN(C(c3c(C)n[nH]c3)=O)CC2F)c(F)cc(Br)cc1F 43853,C(CCO)(C(=O)O)NC(=O)Nc1ccc(Cn2ccnn2)cc1 43854,n1(CC)cnc2c(NC3CCCN(C(=O)Cn4ncc(Cl)c4C)C3)ncnc12 43855,C#CCCCC(C)C(=O)Nc1c(C)cnn1C.C1(C(=O)N)(Cc2c(C)ccs2)CCC1 43856,Cc1cc(C(N2CCC(CN(C)C(C3CCN(C)C3)=O)C2)=O)cnc1C(F)(F)F 43857,C12(C(=O)NCC(CC=C)NC(=O)COC3CCCC(C)C3)COC(CF)(C1)C2 43858,Cc1cc(Cl)c(C(=O)NCC2(CNC(C3C(C)C3(F)F)=O)CCC2)s1 43859,CC(N=c1ccnc(NCCOc2ccc(F)cc2Cl)[nH]1)c1nncs1 43860,CC1=NOC(C)(CC(=O)NCc2c(C(=O)OC(C)(C)C)cnn2C)C1 43861,c1(C(C(=O)N(C2CCN(C(=O)C=COCC)CC2)CCC)(F)F)cc(C)ccn1 43862,c1(CCN(C(=O)CCCN(C)C(C2C=CCCC2)=O)C)nccc(O)n1 43863,c1(C(N2CCC(COC)(NC(C3CC=CCC3)=O)C2)=O)ccc(OC)c(Cl)n1 43864,c12ccccc1NC(=O)NC2CNC.C(C(O)CO)OCC 43865,N1(C(c2ncc(C)cc2F)=O)CC2CCC(N(C)C(c3occc3C)=O)C2C1 43866,C1(CNC(C2(OC)CCC2)=O)CC(C)(C)CN1C(=O)CC1CC(OC)C1 43867,C(=O)(CCS(C)=O)NC(c1ccccc1)CNC(C1C(OC(C)=O)C1)=O 43868,C1(NC(C2C(CNC(C(COCC)C)=O)CCO2)=O)CNC(=O)C1(C)C 43869,C(CCCCC(=O)N(C)CCOCCNC(C1CCC(C2CC2)C1)=O)SC 43870,c1(OCC)ccc(C)c(C(=O)NCC2CC2NC(c2nc(C3CC3)oc2C)=O)n1 43871,C(=O)(CC(C(F)F)c1cccc(F)c1)N(CC(C)N(C(C=C(C)Cl)=O)C)C 43872,CC1(C)C(CNC(=O)CN2CCC(c3nn(-c4ccccc4)cc3F)C2)CC1O 43873,Cc1cc(C(=O)NCCCC2CCN(C(=O)CC34CCCC3C4)CC2)c(O)nn1 43874,N1(C(C(C(C)C)OCC)=O)CC2CCC1C(NC(=O)Cc1n[nH]c(C)n1)C2 43875,N1(C(c2c(C(C)C)onc2)=O)CCC2(CC(C(=O)NCCN(C)C)C2)C1 43876,C1(OCC(N2C(C3(NC(c4cc(F)c[nH]4)=O)CC3)CCC2)=O)CCCCCC1 43877,C1(NC(Cn2nnc(=N)[nH]2)=O)CCCCCN(C(C23CCN(CC2)CC3)=O)C1 43878,c1(OC)c(C(=O)NC2CC(NC(=O)C(C(C)C)NCC(C)C)C2)cc(Cl)cc1C 43879,N1(C(c2ccc(C)cc2)C(=O)NC(CC)(C)C)C2CCC1CC(F)C2 43880,c1(NC(C2CCCCN2C(c2cc(Cl)c(Cl)cc2F)=O)=O)cc(F)c(O)cc1Cl 43881,CC1CN(C(=O)COC2CCN(C(=O)C=CCCC(C)C)C2)CC(C)(C)O1 43882,Cn1nc(C2CC2)cc1CC(=O)NC1CN(C(c2cncc(F)c2)=O)CC1F 43883,c1(NC(CN2CC(C)C2)=O)ccnc2c1cnn2C.C12CN(C1)C(=O)CO2 43884,N1(C(C2(C)N(C(C(CC)N(CC)CC)=O)CCC2)=O)CC2CC(NC)C2C1 43885,N1(C(=O)Cc2cc(F)cc(Cl)c2)CCC2OCCN(C(=O)C=CCO)C2C1 43886,C1(CNC(C2N(C(C)=O)CC(O)C2)=O)CC2CCC(C1)N2C(=O)COC1CCC1 43887,C1(C(N(C)CCC2OCCO2)=O)CCN(C(c2cc(Cl)cnc2F)=O)CC1O 43888,c1(C(N(CC(C)(C)CNC(C2(C3CCCCO3)CC2)=O)C)=O)cc(CN)nn1C 43889,C1(C(=O)NC2CCCC(CN(C)C(c3ccncc3O)=O)C2)OCCOC1(C)C 43890,CS(=N)(=O)CCNC(=O)C(Cc1cc[nH]n1)NC(=O)CC1CCSC1 43891,N1(C(C(C=C)O)=O)C2CCC1CN(C(c1sc(Cl)cc1Cl)=O)C2 43892,CC1CN(C)C(=O)CN1S(=O)(=O)c1ccc(C(=O)O)s1 43893,C(N=c1[nH]c(=NCC2CCC=CO2)c2cccc(F)c2[nH]1)c1cn(C(C)C)nn1 43894,C#CCC(C(=O)NCCCOCC1CC1)NC(C1CC=CCC1)=O 43895,C1(CC(=O)NC2C(NC(CSCC=C)=O)C2)OCCCC1(C)C 43896,C(=O)(C(O)C(F)(F)F)NC1CC2(C(C(N3CC(C)(OCC)C3)=O)C2)C1 43897,N1(C(COc2c(CC)cccc2)=O)CC2CC1CN2Cc1csc(Br)c1 43898,C1(C(=O)NCC#CCNC(c2cc(C)n(C)c2)=O)CC(c2cccc(F)c2)=NO1 43899,c1(C(=O)NCC2C(C(N3CCC(CC#C)C3)=O)C2)cccc2nccn12 43900,c1(CC)ccc(C(N2CCC(N(C)C(c3cnc(O)cc3OC)=O)C2)=O)c(Cl)c1 43901,c1(C(=O)NC(c2ccccc2)CCC)ccc(N2CCC(N)CC2)cc1 43902,O(NC(=O)C(C)(C)S(C)(=O)=O)C(CC(C)C)C(=O)N1CCCNC(=O)C1 43903,n1(CCCNC(C2CC(n3cc(N(C4CC4)CC4CC4)nn3)C2)=O)cnnc1O 43904,c1(N(C)C)ccc(NC(N2CCC(O)(C(F)(F)F)C2)=O)nc1 43905,N1(CC(=O)NC(CC)(C)C)CCC2(CC1)CC2(C)C(=O)NC1CCCN1CC 43906,C1(C(N(CC#C)C)=O)CC12CCN(C(=O)CN1CC(C)(C)C1)C2 43907,C(c1cccnc1)=C(C)C(=O)NC1C=CCCC1C(=O)NC12CC(C1)C2 43908,C1(NC(c2ccc[nH]2)=O)CN(C(C23CCC(CC2(F)F)C3)=O)Cc2nccn2C1 43909,CCCCCC(F)C(=O)N(CC(N1CC(O)CC1COC)=O)CC1CC1 43910,c1(C(=O)NCC2C(C)C2NC(C2CC(=C3CC3)C2)=O)ccc2[nH]nc(O)c2c1 43911,C1(F)(CNC(C2C(CC(C)(C)C)C2)=O)CCN(C(=O)CS(N)(=O)=O)C1 43912,CC(=O)CCN=C(NCc1ccn(C)n1)NCC12CCCC(C1)OC2 43913,Cc1nn(CC(N2CCC(C(F)CNC(c3ccoc3)=O)CC2)=O)cc1Cl 43914,N1(C(C=CC)=O)CCC2(CC1)CN(C(=O)C(C)n1cccn1)CC2CO 43915,c1(C(N2CCC(CCNC(C3C(=C)C3)=O)CC2C)=O)ccc2nnc(O)n2c1 43916,C1(CNC(CC2C(OCC)COCC2)=O)CN(C)CCN1C(C1CNC(=O)N1)=O 43917,C(=O)(C#CC1CC1)N1CC(CC(C)NC(c2c[nH]nc2-c2ccccc2)=O)C1 43918,C(=O)(C(S(C)(=O)=O)C1CC1)NCC(C)CNC(C1(C)CCSCC1)=O 43919,CC1COC2(CCC2)CN1C(C1CCN(C(c2cc(C3CC3)no2)=O)CC1)=O 43920,N1(C(CC(C=C)(C)O)=O)CCC2(C1)CN(C(=O)Cc1c(C)cnn1C)CCO2 43921,C(=O)(C(CC(C)C)NC(=O)OC)NCC(C1(OC)CCOCC1)(F)F 43922,C1(C(N2CC(CC(=O)NCCc3cc(C)n(C)n3)OCC2)=O)CN2CCN1CC2 43923,c1(C(N2C(C(=O)NCc3ccc(C(C)C)cc3)C(O)CC2)=O)ccc(Br)c(Cl)n1 43924,CCCC(C(=O)NC(C)(C)CNC(c1cccc(COC)c1)=O)S(N)(=O)=O 43925,c1(CC)nnc2cc(NCC3CN(C(=O)C(C)Cc4ccco4)C3)ncn12 43926,C1(O)(CCNC(CC2CC(=C)C2)=O)CCN(C(c2cnc(C3CCCO3)s2)=O)C1 43927,c1(C(C(=O)OCC2CCC(F)(F)C2)OC)cccc(CC(F)(F)F)c1 43928,C(=O)(C1=CC2CCC1C2)NCC(C)NC(c1ccc(Br)cn1)=O 43929,c1(CNCC(O)C(F)(F)F)c(O)ccc(F)c1F 43930,CCC(=O)CCC(=O)N1CCOCC(CNC(c2sccc2OCC)=O)C1 43931,C(CCCCC(=O)NCC1CCN1C(c1sccc1Br)=O)OCC 43932,C1(C(N2C(CCC(=O)NCC(CC(C)C)O)CCC2)=O)CCN(C)C(=O)C1 43933,N1(c2ccc(NCC(=O)Nc3cc(F)cc(F)c3)cc2)CCc2sccc2C1 43934,C1(C)(NC(CCCNC(C)=O)=O)CCC(NC(C2(O)CCSCC2)=O)CC1 43935,C(=O)(C1CC(=O)c2ccccc21)N1CCC(NC(=O)Cn2cnnn2)(CF)C1 43936,CN1CCC(NC(C2N(C(c3ccc(O)cn3)=O)CCC2(C)C)=O)C(C#N)C1 43937,CCC(C)C(C(=O)NC1CCN(C)CC1C)N(C(=O)CCC1CCC1)C 43938,Cc1ccc(C)c2[nH]c(C(=O)NCC3CCC3NC(C3CCS(=O)CC3)=O)cc12 43939,c1(C(=O)NCCCCNC(=O)CCc2cncnc2)c(Cl)ccc2c1OCO2 43940,C1(C(C(CC=C)=O)=O)CCCN(C(=O)NC(C2(NC3CC3)CCC2)=O)C1.C1(N)CC1 43941,c1(C(=O)NC2(CC=C)CN(C(=O)C=CC(C)C)C2)cc2c(s1)COCC2 43942,C1(C)(C(=O)OC)CC(C(=O)N(CC(O)CN(C)C(c2coc(Cl)c2)=O)C)C1 43943,c1(CN(C)C(=O)NC2(c3cccs3)CCC2)cnn(C)c1N 43944,C1(CNC(C2C(C)=CCS2)=O)CN(C)CCN1C(=O)C1=CC(C)C1 43945,c1(OC)ccc(CN(C)CC2CCCN(C(C3CC(C)(C)C3)=O)C2)cc1C 43946,C1(C)(CC)CC(C(=O)NC(c2cccnc2)c2nc(C)cs2)CCO1 43947,CCCCCC(F)C(=O)NC(C1CCCCCC1)CNC(c1cncn1C)=O 43948,c1(C(=O)NCc2cccc(CNC(C=CSC)=O)c2)ccc(C(C)(F)F)nc1O 43949,C1(CC(=O)NCCN(CC(C)O)C(c2cscc2F)=O)CCC(C)(C)CO1 43950,c1(C(=O)NC2C(CC)CN(C(c3cccnn3)=O)CC2)cccc2nccn12 43951,c1(C(N(C(C)CNC(C2(C(F)(F)F)CCCC2)=O)CC)=O)ccnnc1 43952,c1(C(=O)NCCN(C(C)C)C(C2(C)CC=CCO2)=O)cc2ccc(O)cc2n1C 43953,C1(O)(CS(=O)(=O)NC(C(C(C)C)NCCOC2CCCC2)=O)CCCCCC1 43954,c1(C(=O)OCC)cnc(N2CCS(=O)C(C)C2)cc1C 43955,C1(NC(C=CC(C)C)=O)CC(NC(=O)Cc2ccccc2)CC1O 43956,N1(C(CNC(CCC(C)C)=O)=O)CCC2(NC(=O)CC(=O)N(C)C)CC2C1 43957,C1(OC)CC(CNC(c2cc(C(C)(C)C)nn2C)=O)N(C(c2nn[nH]c2Cl)=O)C1 43958,N1(c2nnc(C)o2)CCC(C(C)NC(C2C3COCC23)=O)CC1 43959,c1(NC(=O)NOc2ccc(Cl)cc2)cnc(Br)cn1 43960,CC(C(=O)N1CCCC1C1(O)CN(C(C2C3CCCCCC23)=O)C1)S(N)(=O)=O 43961,c1(C(N2CC3C(NC(=O)CO)CC(C3)C2)=O)n[nH]c2ccc(Cl)cc12 43962,Cc1cnc2cccc(C(N3CCC(NC(=O)Cc4cnc[nH]4)C(O)C3)=O)c2c1 43963,C1(CN(C(C2C(C)CCC2)=O)C)COCCN1C(C1CC(=O)N(C)C1)=O 43964,C(=O)(C(C)(CO)CO)N1CCCC(C(=O)Nc2c(C(C)=O)cccn2)C1 43965,c1(C(=O)NC(C)CCNC(=O)CC(C)N(C)C)ccc2nccnc2n1 43966,C(CCC(N)=O)(C(=O)NCC1CCCCN1C(=O)C(O)C(F)F)NC(C)=O 43967,Cc1ccc(C2(C(=O)NCCNC(C3(C)COC3)=O)CC2)c2ccccc12 43968,C1(NCC2CC(OCC)C2)CCS(=O)(=O)C(C)(C)C1 43969,N1(C(C2CC(SC)C2)=O)CC(C(=O)NC2CC2)CCC1C 43970,N1(c2n(CCOCCOC)nnn2)CCC(O)(CN2C(=O)CN(C)C2=O)CC1 43971,c1(C(N2CCC(CNC(C=CC=CCC)=O)C(C)C2)=O)cc2c(cn1)CCCC2 43972,O=S(=O)(c1cnccc1N1CCCC(CCO)C1)NCC1(CC2CC2)CC1 43973,C1(F)(CNC(C(CSC)OC)=O)CCN(C(=O)CC2CC(=O)C2)C1 43974,C1(c2n(C)cnc2)COCCN1C(=O)CCC1CCCCO1 43975,c1(C(N2CCN(C(c3scc(C)n3)C(=O)NC3CC3)CC2)=O)cc(C)cc(C)c1N 43976,CC(CC(F)(F)F)C(=O)N1CCN(C(=O)CCCN2CCCC2)C(C)C1 43977,c1(C(=O)NCC(C)(C)NC(=O)Cc2ccoc2)ccc(-c2ccccc2)s1 43978,N1(CC#N)CCCC(NCc2ccc(I)cc2)C1 43979,c1(C(=O)NC2CC(C)N(C(c3cc4cccnn4c3)=O)C2)ccc2nonc2c1 43980,c1(C(C)=O)ccc(C(=O)NCC2(CN3CCN(C)CC3)CC(F)(F)C2)cc1Cl 43981,CC1(C)C(CC(=O)NC2CCC(NC(c3coc(Cl)c3)=O)CC2)CC1O 43982,Cn1cc(S(=O)(=O)CCNC(=O)Cc2ccn(C)c2)cn1 43983,C(C(C)(C)C#CC(=O)NCC(c1ccnn1C)O)NC(CN1C(C)CCCC1)=O 43984,C=C(C)C1OCCC1C(N1CC(C(C)NC(=O)Cc2cnc(C)s2)C1)=O 43985,C1(C#CC(=O)NCC2CC2CNC(=O)CCCCN(C)C)(CC)CC1 43986,C1(C(=O)NCC(S(C)(=O)=O)CNC(C2CCCCC2O)=O)OCC2COCCC12 43987,C=CCCCC(C)(C)CN=c1[nH]c(C)cc(=NCC2(C)CSCCO2)[nH]1 43988,C(=O)(C(F)C(=O)NC(C)CN(C(C1CSCN1C(=O)NC)=O)CC)OCC 43989,N(C(=NCCOCC)N1CCC2(CCCCCC2)C1)C(C#C)CC 43990,C1(NC(C2C(C(C)NC(=O)CCc3ccc[nH]3)C2)=O)CCCC(O)CC1 43991,c1(C(=O)NC2CN(C(C(OCC)OCC)=O)C(C)(CC)C2)n[nH]c(C)c1[N+](=O)[O-] 43992,c1(C(=O)NC(CNC(CSC)=O)C2CCC2)cnns1 43993,C(C(F)(C(=O)NCc1ccnc(Cl)c1)C(C)C)NC(c1c(C(C)C)c[nH]c1)=O 43994,C1(O)(C(C)CNC(=O)COC(F)F)CCN(C(c2c(Br)ncn2C)=O)C1 43995,Cc1cc(C(=O)NCC#CC(=O)N(C)CC2CC2(F)F)ccn1 43996,C(=O)(C1CCCc2c1ncn2C)N1CCCCC(NC(CCCC#C)=O)CC1 43997,C1(C(=O)NCCCCN(CC)CC)C=CCN(C(=O)C(=O)N(C)C)C1 43998,C1(NC(c2cc(C)[nH]n2)=O)CCCOC12CCN(C(C1COC(=O)C1)=O)CC2 43999,N1(C(C)=O)CC(C)CN(C(=O)CCNC(C2(CC=C)CCCC2)(C)C)C(C)C1 44000,c1(CN2C(C(=O)NC(C3CCCCC3)CC)C(O)CC2)ccccc1[N+](=O)[O-] 44001,C(N=c1cc(NCc2cnn(CC(F)F)c2)nc[nH]1)c1nc(C(C)C)sc1 44002,c1(C(N2CCN(C(c3ccn(COC)n3)=O)C3C2C3)=O)cn2c(C)cccc2n1 44003,C1(CC(=O)NC2CC(CNC(CSC)=O)C2)CSc2ccccc2O1 44004,c1(CN2C(C(=O)NCC3CCCO3)C=CC2)ccc(Cl)c(O)c1 44005,c1(N2CCC(CCOC)(OC)C2)nc(Cl)nc(-c2ccccc2)c1C 44006,N1(C(C(C)CC#N)=O)CC2CCC(CN=c3nc[nH]s3)(C2)C1 44007,C1(C(=O)NCCC(CNC(C2CC3(CCC3)C2)=O)O)CC2CCC1C2 44008,Cc1cccc(C(=O)NCC2CCC2C(=O)NC(C)(C)CNC(N)=O)c1 44009,C1(CN(C)C)CCCC1C.CC1CN(C)C(=O)C=CC(=O)N1 44010,CCC(CCC(=O)N1CCCCC1CO)NC(c1cc(C)ncn1)=O 44011,C1(CNC(C2(C)CC2(F)Cl)=O)C2CN(C(c3ccn(C4CC4(F)F)n3)=O)CC12 44012,C=Cc1ccc(C(N2CCCC(C)(CNC(c3c(Cl)noc3C)=O)C2)=O)cc1 44013,CC1(C)C2CC(C(=O)NCC3CC(F)(CNC(C4CCS(=O)(=O)N4)=O)C3)CC12 44014,CCC(C)C(=O)NCC(N1CCCC1C(=O)NCc1ccn(C2CCC2)n1)=O 44015,c1(C(=O)NC(CN(C(c2cnn(CC)c2Cl)=O)C)C)cc(O)nc(C)n1 44016,CC(CNC(C1CC1Cl)=O)C(F)C(=O)NCCCN1CCOCC1 44017,c1(C(=O)NCC(CC)NC(=O)Cn2ncccc2=O)ccnc(S)c1 44018,C1(CCNC(CCC=C)=O)CN(C(=O)C(CCC)OCC)CCCO1 44019,c1(C(=O)NCC2CN(C(c3c(C)coc3C)=O)C(C)(C)C2)cc(P(C)(C)=O)cs1 44020,C(C(N=c1cnc(C(N)=O)c[nH]1)c1n(C)ncc1)NP(C)(C)=O 44021,N1(C(C=C(C)C(F)F)=O)CCC(C2CC2)C1C(=O)NCC(CC1CC1)CO 44022,C(C(CC(C)C)C(=O)NCCOC1CN(C(C2(OC(C)C)CCOC2)=O)C1)OC 44023,CS(=O)C1(CNC(=O)NCC2CNC(=O)C2)CCC1 44024,c1(C2(C)CN(C(=O)NCCCc3nccc(C(F)(F)F)n3)C2)ccccc1Br 44025,C1(C(=O)NC(C(=O)NCc2ccc(C)o2)CC2CCC2)CCCC(=O)C1 44026,c1(C(N2CC(c3nncn3C)C2)=O)ncc(F)cc1F.CN1CCC2(C1)C(=O)N2 44027,C1(C(=O)NC2CC2NC(=O)C(F)(F)C2CCOCC2)(OC)CCSCC1 44028,c1(OC)c(F)ccc(C(=O)NCCN(C(C2CCCCC2)=O)C(C)C)c1F 44029,c1(CC(=O)NC2CCN(C(COCCC)=O)C2)ccccc1CS(N)(=O)=O 44030,Cc1cc(C(N2CCC(NC(C3CC34CCCC4)=O)C(CO)C2)=O)ncc1CO 44031,C1(COC)CN(C(c2nccc(Br)c2C)=O)CCN1C(C1CC2CC2C1)=O 44032,c1(C(N(CCCC(=O)NCCCc2cc(C)no2)C)=O)n[nH]c2c1COC2 44033,Cc1nc2ccccc2n1CCC(=O)NCCC(C)NC(=O)C1=CCCC1 44034,C1(CCC#C)NC(=O)N(C(c2nn(C)cc2O)C)C1=O 44035,C1(C(N2CCC(C#N)C2)=O)(CC)CCN(C(=O)COC(C)=O)C1 44036,c1(C(=O)NCc2ccc(C(=O)NC(C=C)(C)CC)s2)cncc(Cl)c1 44037,CC1C(NC(=O)CS(N)(=O)=O)CCCN1C(c1cncc(C(C)(F)F)c1)=O 44038,C1(C(N2CCC(C(C)(C)O)CC2)=O)(CCc2cc(Br)c[nH]2)CCCN1CC 44039,N1(C(C2(NC(=O)C3=CCCC3)CC(CO)C2)=O)CCn2nncc2C1 44040,c1(CSC)cc(C(=O)NCC2CC(NC(C3CCN(C(C)=O)C3)=O)C2)ccc1F 44041,N1(C(C(CC=C)NC(=O)CN2CCCCCC2)=O)CC(C2CC2(F)F)C1 44042,C(CC1CCC1)(C(=O)N(CC(C)NC(=O)Cn1cnnc1O)C)NC(C)=O 44043,NS(=O)(=O)c1ccc(C(=O)NCC2CCCCC2NC(=O)CC2NC(=O)NC2=O)o1 44044,Fc1cc(C(F)(F)F)ccc1C1CC1c1cccc(Br)c1 44045,C12(CNC(C(CNC(=O)C#CC(C)C)OC)=O)CCC(F)(CC1)C2 44046,C(=O)(C(C)P(C)(C)=O)N(CCN(C(C)C)C(c1ncccc1OC(F)F)=O)C 44047,C1(C(C)N(C(=O)C(N(C)C)N(C)C)C)CCCN(C(=O)OC(C)(C)C)CC1 44048,C(CC(C(=O)N1CC(C)(CO)C1)NC(=O)CCc1cccs1)OCC 44049,c1(C(N2CCC(NC(C(CCSC)(C)C)=O)C(C)C2)=O)cc([N+](=O)[O-])cc(C)n1 44050,C(CC1CCOc2ccccc21)n1cc(C(=O)Nc2c(C#N)cccn2)nn1 44051,C1(NC(C=C(C)c2ccsc2)=O)CS(=O)(=O)CC1NC(=O)CCc1csc(C)n1 44052,c1(C(=O)NCC2(F)CCC(NC(CC(CC)OC)=O)C2)c(C)nc(O)nc1C 44053,Cc1c(C(=O)NCCNC(C2OCCC2C(F)(F)F)=O)c(=O)oc2ccccc12 44054,Cc1cc(C(=O)N(CC(=O)NC2CC3CC4C(C3)C24)C2CC2)c(C)nn1 44055,c1(CC(=O)NC2(COC)CCN(C(=O)CCC#N)C2)cc(F)cc(Cl)c1 44056,N1(C(C(C(C)C)SCC)=O)CC(CNC(c2cnc(O)c(C)c2)=O)C(C)(C)C1 44057,C12(CNC(=O)C=Cc3cccnc3)CCCC1N(C(=O)C=CC1CCCC1)CC2 44058,C1(NC(c2cc(C)on2)=O)CC1C1CCCN(C(=O)CN2CCN(C)CC2)C1 44059,N1(CC(c2ccc(CN(C)CC)cc2)=O)C(=O)c2cccnc2C1=O 44060,N1(C(C2CC(C)=C(C)CC2)=O)CC2(CCCC(CNC(=O)Cn3nccn3)O2)C1 44061,S(=O)(=O)(c1ccc(NCc2nncn2C(C)(C)C)c(F)c1)N(C)Cc1cscn1 44062,C1(C(C(=O)N(CCNC(=O)C(c2ccn(C)c2)C)C(C)C)OC)CCCCCC1 44063,c1(C(=O)NC(CNC(c2c(C)ccc(SC)c2)=O)C2CC2)ccc2c(c1)CCO2 44064,C1(CC)CCN(C(=O)CC=CC(C)(C)C)C1C(=O)NCCc1nncs1 44065,N1(C(=O)OCC)CCCN(C(CC2CC2)C(=O)NC)CC1 44066,C1(NC(=O)CC(F)(F)C(F)F)CC(NC(c2csnn2)=O)C12CCOCC2 44067,C1(CN(C(CSCC(C)=O)=O)C)CCCCN1C(=O)Cc1csc(S)n1 44068,C1(NC(c2cn(CCC)nn2)=O)CCN(C(=O)C(c2ccc(F)cc2)CC)CC1 44069,C(=O)(C1COc2ccccc21)N(C1CCCN(C(C2(CF)COC2)=O)C1)C 44070,c1(C(C)NC(c2n(CCCOC)nnn2)c2cc(OC)ns2)cccc(OC)c1 44071,CC(C)(C)C(CNC(C1CCC=CO1)=O)NC(=O)CCN1CCOCC1 44072,C(=O)(CCC(=O)NC1CC(CNC(C2CSCN2C(C)=O)=O)C1)NCC 44073,C(=O)(C1=NN(C)C(=O)CC1)NCCC(C)N(C(c1cncc(C)n1)=O)C 44074,C(C(=O)N1OC2C=CC1CC2)(C1(O)CCCCC1)NC(C(C)C1CCCC1)=O 44075,c1(OC)ccc(CC(=O)NCCOCCNC(c2cc(Cl)ccn2)=O)nc1 44076,NC1C2CCC1N(C(c1ccnc(OCCO)c1)=O)C2 44077,c1(C(CNCC23OCC(C(C)C)(C2)C3)O)ccc(S(C)(=O)=O)cc1 44078,c1(C(=O)NCC(C)(C)NC(c2c(CC)n(C)cc2)=O)oc2ccc(C)cc2c1C 44079,c1(C(N2CCC(=CCNC(CC(C=C)CC)=O)CC2)=O)n[nH]c2c1CC1CC21 44080,C(=O)(C(CCc1ccc(F)cc1)C(C)(C)C)N(C(C1C(OCC)C1)=O)C1CC1 44081,c1(SC)ccc(C(=O)NCC(C(C)(C)C)NC(C2CCCCC2)=O)c(Cl)c1 44082,c1(CCNC(N2CCN(C(C)=O)C3C2CC3)=O)ccc2cc(OC)cc(Br)c2n1 44083,c1(C(N2CCOCC(CNC(C(C(=C)C)(C)C)=O)C2)=O)c([N+](=O)[O-])cnn1CC 44084,CC1=C(C(=O)NC2(COC)CCN(C(C3(c4ccccc4)CC3)=O)C2)CCC1 44085,O=C(C1=CCCCC1)NCCCN(C(c1cccnc1)=O)C1CC1 44086,S(=O)(=O)(c1ccc(N2CCCCC(C)(F)C2)c(C#N)c1)NCc1cc(CC)no1 44087,C1(C)(C(=O)NCCCCNC(c2c(OC)c[nH]n2)=O)CCC(C(F)(F)F)CC1 44088,C=CC(C)CC(=O)NC1CC(CNC(c2ccsc2-n2cnnn2)=O)C1 44089,CC(C)C(CNC(c1cnn2c1OCC2)=O)C(=O)NCCCc1cnccn1 44090,n1(CC)nc(C)c(C(=O)N(CCCCNC(=O)COCc2cccnc2)C)c1Cl 44091,C1(NC(c2ccc(C(C)=O)o2)=O)CCN(C(=O)CCc2cncs2)CC1C(C)C 44092,c1(C(N2CCC(CC(=O)Nc3cnc(C4CC4)nc3)CC2)=O)cnn2c1CCC2 44093,C1(C(=O)NC(CCSC)C(=O)NC(C)(C)CCCN(C)C)CN(C)CC(C)O1 44094,N1(C(c2cc(C)sc2)=O)CCN(C2CCCN(C(=O)CCOC(C)C)C2)C(=O)C1 44095,C1(C(=O)NCCCn2ccnc2)CCC2(CC2)N1C(=O)C=CCN1CCCC1 44096,c1(OC)nn(C)cc1C(=O)NC1CCC(CNC(=O)C(C)n2cccn2)CC1 44097,C(=O)(C(C)C(C)NC(c1c[nH]nc1OC)=O)N(CC(=O)OC)C1CC1 44098,N1(C(C(CC=C)OC)=O)CCC2(CCC(NC(=O)Cc3ccccc3C)CC2)C1 44099,c1(NC(C2(C3N(C(C(CC)CC)=O)CCC3)CC2)=O)ccc(F)cc1SC 44100,c1(OC)cccc(C(c2nnnn2C2(C)CC2)NCc2cn(C)nc2C(C)C)c1 44101,c1(C(=O)NC(C)CCNC(=O)C(O)c2cnc[nH]2)ccc(Cl)o1 44102,c1(C(=O)NCC(C)NC(c2ccn(C(CC)CC)n2)=O)cc(C)nn1CC 44103,N1(C(C(CC(=C)C)C)=O)Cc2ccccc2C(NC(=O)Cc2ccc(C)o2)C1 44104,c1(C(C(N2CCC(O)(CNC(C3C(COC)C3)=O)C2)=O)(C)C)cccc(C#N)c1 44105,c1(NC(c2n(CCCOC)nnn2)(COC)C2CCCC2)ccc2nncn2c1 44106,c1(C(=O)NCC(C)N(C(CCC(C)c2ccccc2)=O)C)cnc2[nH]cnc2c1 44107,C(=O)(C1=C(Cl)CCOC1)NCCC(C(=O)Nc1c(OC)cc(F)cc1)(C)C 44108,C1(C(N2CC(COC)(NC(=O)Cc3cc(C)on3)C2)=O)CC=C(C)CC1.OC 44109,N1(C(C(CCC)(C)C)=O)CCC2(CCN(C(=O)CC3CCCCC3(F)F)C2)C1 44110,N1(C(C(C=C)O)=O)CCC(C(=O)N2CCC23CCCCC3)=C(F)C1 44111,C(=O)(CC(C)CC(C)(C)C)NC1(C(=O)NCCC#C)CCN(C)C1 44112,C1(C(=O)NCC(CN(C(c2c(C)cc(C)o2)=O)C)O)CCC(C2CC2)CC1 44113,Cc1nc(C(C)C)ccc1C(=O)NCC(O)CCNC(c1cc(F)cc(F)c1)=O 44114,CC1CCN(C(=O)C2=CCCCC2)CC1CNC(=O)C=Cc1ccoc1 44115,Cc1cc(N2CCn3cccc3C2)nc(=NCCCc2ccc(C)c(C)c2)[nH]1 44116,C#CCC(C)(C)C(=O)NCC(C)N(C)C(C1CC1C#N)=O 44117,N1(C(C(COCC)N(C)C)=O)CCCC(Cc2ccc(OC)cc2)C1 44118,c1(C(=O)NCCNC(C2CCN(C(CC)=O)C2)=O)nnn(C2CCOC2)c1C 44119,c1(-c2ccc(C(=O)NC3C(C)(C)C3)cc2)ccc2c(n1)CCC2=O 44120,c1(C(=O)NC2CN(C(C3CC3(Cl)Cl)=O)CC2C(F)F)oc2ccccc2c1CO 44121,n1(CC)c2ccccc2c2cc(-c3nc(CC4CC4)nn3C(C)C(C)C)ccc12 44122,Cn1ncc2nc(Cl)nc(NCC3(N)CCCC3(C)C)c12 44123,C1(O)(C(=O)NC2CC3(C(NC(c4c(C)c(N)ccc4)=O)C3)C2)CCCC(C)(C)C1 44124,C1(N=c2cc(Br)n(C)[nH]2)(c2n(CCCSC)nnn2)C(C)CCC1 44125,c1(C(=O)NCCSC)cc2cc(-c3cn(C)nc3C)ccc2oc1=O 44126,C1(NC(c2cccc(NC(C)=O)c2)=O)CC(C)CN(C(C2CCC(C)(C)O2)=O)C1 44127,C(=O)(C(C)C(=O)N1CCN(CCCNC(=O)C(C)(C)n2cnnn2)CC1)OC 44128,c1(C(=O)NCC2N(C(C(COC)O)=O)CCOC2)c(Cl)cc(Cl)cc1Cl 44129,C1(C)(C(=O)NCCCN2CCN(C(CCSC)=O)CC2)C(C)(C)C1(C)C 44130,C1(C(N2CCC(OC(C)=O)C2)=O)CCN(C(=O)C(C)(C)CO)CC1(C)C 44131,c1(C(=O)NC2CC(N(C(C(CC=C)OC)=O)C)C2)[nH]nc2ncccc12 44132,c1(C(=O)NC2CCCCN(C(C3C(CCC)CCC3)=O)C2)cccc2[nH]ccc12 44133,CC1(C)CC(=O)NC1CSCC(CO)SC(C)(C)COC 44134,c1(CCC(=O)NCCCC(=O)NCC(CC=C)NC(N)=O)ccc(Cl)c(OC)c1 44135,C1(C(=O)NC2CC(C(C)C)OC2)C=CCN(C(=O)Cn2ccnc2)C1 44136,c1(C(=O)NC2CC(CCC(N3CCC(OC)CC3)=O)C2)ncc(F)cc1C 44137,c1(C(=O)NCCCN(C(=O)CC2C=CCCC2)CC)cc(C(F)F)cs1 44138,Cc1nc2ccc(C(C)NC(c3cc(Cl)ccc3C(F)(F)F)C)cc2o1 44139,N1(C(c2ncc[nH]2)=O)CCC(C2CCCN(c3nccn4nnnc34)C2)CC1 44140,C#CC1CC(CONC(=O)C2CC2CCC)C1 44141,C#CC1(C(N2CC(C(C)(C)C#N)C2)=O)CN(C(c2cc(OC)ccn2)=O)C1 44142,c1(CN(C(C2(CNC(c3nc(Cl)cs3)=O)CCC2)=O)CC)ccncc1 44143,N1(C(CCC=CC)=O)CCC2C1CCCN2C(C12CC(c3ccccc3)(C1)C2)=O 44144,c1(NC(C2=NOC(C)C2)=O)cccc2c1CN(c1ccccn1)C2 44145,c1(C(C)=O)ccc(C(=O)NC2CN(C(=O)C(c3cccc(O)c3)C)CC2C)cc1 44146,CCN=c1ccc(C(=O)NC2CC2NC(c2cc(CC(C)C)c[nH]2)=O)c[nH]1 44147,C1(C)(c2nc(CC)on2)CCN(N2CCC(C)(NC(C)=O)C2)C1 44148,C1(NC(C(C2CCCN(C(=O)CSC3CC3)C2)(C)C)=O)CCOC2(CCC2)C1 44149,C(=O)(C1CCc2nccn21)NCC(C1CCN(C(C2(C(C)C)CCC2)=O)CC1)F 44150,C1(NC(=O)CCCF)CN(C(c2cccc(F)c2)=O)CC1C(F)F 44151,N1(C(Cc2c(C)n[nH]c2C)=O)CC(NC(c2cc(CO)ccc2O)=O)C(C#N)C1 44152,C(c1cccc(CO)c1)=CC(=O)NC1CC1NC(=O)Cc1c[nH]nc1O 44153,N1(C(c2c(CC)ccc(F)c2)C(=O)NCCC2CC2)CCC2OC(=O)OC2C1 44154,c1(C(c2cccnc2)C)noc(C(C)C(=O)NC(=O)CCCN)n1 44155,c1(C(=O)NC(C2CCCC2)CC)cc(CNC(C2CCC(F)CC2)=O)nn1C 44156,C1(C(N(C(C#C)C)C)=O)CN(C(=O)Cc2scnc2C)CCO1 44157,c1(C(=O)NCCCNC(C(C)C2CC2)=O)ccnn1-c1cccnc1 44158,C(=O)(CCCc1nccs1)C(C=CCNC(=O)OCC1(NC(C)(C)C)CCC1)=O 44159,CC1CC(C)N(C(c2oc(S(N)(=O)=O)cc2C)=O)CCN1Cc1ccccc1 44160,C(=O)(CCCCCCNC(=N)N)N1CCCC(c2nnc(C)o2)C1 44161,n1(CCCNC(C2(CNC(C(C3CC3)OCC)=O)CCC2)=O)cc(C)cn1 44162,Cc1cc2ncnc(N3CCC4(CCN(C(c5ccc(F)c(F)c5)=O)C4)C3)c2[nH]1 44163,C12(C(=O)NC3CCN(c4nccc(C#N)n4)CC3)CCCCC(=O)N1CCC2 44164,c1(OC)ccc(CN2CCC(C(N3CCOCC3C)=O)C(O)C2)c(Br)c1 44165,c1(C(=O)NC2C(CNC(=O)C3=CCC3)CC2)ccc2oc(=O)oc2c1 44166,C1(n2cc(CN(C)C(c3cccc(F)c3)=O)nn2)CCCC(F)(F)C1 44167,c1(C(=O)NC(C2CN(C(C3(C)CCCN3C(C)=O)=O)C2)C)ncnc(O)c1Cl 44168,n1(C(C)C)cc2ncc(C(N3CCC4(CC3)CN(C(C3CC3Cl)=O)C4)=O)cc2n1 44169,N1(C(C)=O)CCC2CCC(C1)N2C(=O)CCCCc1ccc(Cl)cc1 44170,CC(C)CC(F)C(=O)N1CC(CNC(c2ccc(O)cn2)=O)C(C)(C)C1 44171,C=Cc1ccc(C(=O)NC(CCSC)C(=O)N2CCC(CC3CC3)C2)cc1 44172,c1(NC(C2C(C(=O)OC)C2)=O)sc2c(c1C(N1CCC(O)C(F)C1)=O)CCC2 44173,N1(C(CC=C)=O)CCCC1C(C(C)C)NC(C1CCC1C(=O)OC(C)(C)C)=O 44174,C1(C(=O)NC(CC=C)C(=O)NC(CCO)C2CCC2)CC2(CCO1)CC2 44175,CC1CCN(C(c2ccn(-c3ccccc3)n2)=O)CC1N(C)C(C1CCCO1)=O 44176,N1(C(C(C(C)C)S)=O)CCn2ncc(CNC(=O)C(N3CCOCC3)O)c2C1 44177,c1(C(=O)NCCCCC(C)NC(c2cocc2C(N)=O)=O)nnc(O)cc1O 44178,C1(CNC(C2(CC=C)CCC2)=O)(NC(C2CCCNC2=O)=O)CCCCC1 44179,N1(C(=O)Nc2cnn(-c3ccncc3)c2)CCCC2(C1)CC(F)(F)C2 44180,CCC(C)(CNC(C1(C)CC1(F)F)=O)NC(=O)CCCn1cncn1 44181,C(CCCCC(=O)NCC1CCCC1NC(c1ccc(C(C)C)cn1)=O)=CC 44182,C12(N(c3cc(C(C)(C)C)c[nH]3)C(C(C)SC)=O)CCOCC1CN(C(=O)C(N)=O)C2 44183,C1(C)(OCC=C)CCN(C(=O)CC(CCC)NC2CCN(CC)C2)CC1 44184,C(=O)(C(O)C(C)(C)C)N(CC(C)O)CCNC(C1CC(O)(CC#C)C1)=O 44185,N1(c2n(CC(=C)C)c(CN3CCCC(O)C3)nn2)CCC(O)CC(C)(C)C1 44186,c1(C(C(N2CCC(C)(CNC(C(CC)C)=O)C2)=O)C)c(C)nn(C)c1C 44187,c1(SC)ccc2c(c1)C(NCC1CC(COc3ccccc3)CO1)CCO2 44188,c1(C(N2C(CNC(CCSCCCC)=O)COCC2)=O)ccc2c(n1)CCOC2 44189,C(=O)(CC(C(F)F)C(C)(C)C)NCC1CC(OC)CN1C(=O)CN1CCOCC1 44190,N1(C(Cc2scc(C)c2)=O)CCC(F)(C(N2CC(CN(C)C)C2)=O)C1 44191,C1(CNC(C2(OC)CCCC2)=O)CC(NC(c2cncn2C)=O)CC1O 44192,C1(C(=O)N(CCCCCNC(=O)CCc2scnc2C)C)(OC)CS(=O)(=O)C1 44193,N1(C(c2c(Cl)ccc(C)c2)=O)CCCC12CCCN(C(c1ccc(=N)[nH]c1)=O)C2 44194,C(=O)(C(C(C)(C)C)NC(C1(C)CC(=O)N(C)C1)=O)N(CCOCC#C)C 44195,C(=O)(C(CC(C)C)C(N)=O)N(C)CC1(O)CCN(C(CC(CC=C)(C)C)=O)CC1 44196,c1(C(=O)OC)ccoc1C(=O)NCC(C)N(C)C(c1csc(C(F)(F)F)c1)=O 44197,C(=O)(C(O)CCS(C)=O)N1CCC(N(C)C(C2(CN(C)C)CC2)=O)CC1 44198,N1(CCOC(CCCOCCOC(C(C)(C)C)=O)=O)C(=O)C2CCCCC2C1=O 44199,C1(NC(CC2C(C)(C)OCC2)=O)CCCC12CN(C(C1CC3C(C1)C3(F)F)=O)C2 44200,O(N(C)C(=O)CNC(C(C)(C)C1CCCO1)c1nnnn1C1CC1)CC 44201,CCC(C)(O)C(=O)N(C)C.N1(CC2(C(=O)O)CC2)CCN(C(=O)Cn2cccn2)CC1 44202,c1(SCC(N2CCC(CCCC(=O)OC)CC2)=O)nc2ccccc2n1C 44203,N=c1nc(N2CC(CC(N)=O)C(CC(N)=O)C2)[nH]c(=NCC2CCCC(=O)N2)[nH]1 44204,c1(C(=O)OCC)cc(F)c(C(=O)NC(C(C)NC(=O)C=C(C)C)C(C)C)cc1F 44205,C1(NC(c2ccc(O)nc2)=O)CC2CN(C(c3ccc(S)cc3)=O)CC2C1 44206,C1(C(=O)NCCc2c(CNC(c3c(C)n(C)nc3)=O)nco2)CCC(O)CN1C 44207,c1(CC(=O)NCC2N(C(CC(C)SC)=O)CCCCC2)ccc2occc2c1 44208,C1(NC(CC(C)(C)O)=O)CCOC12CCN(C(c1cc3ccccc3[nH]1)=O)CC2 44209,C12(C(N3C(C(=O)NC(C)CCCO)CC(F)C3)=O)CCC(CC1)CC2 44210,c1(C(=O)NC(CC(C)NC(COC(C)=O)=O)C)cc(C)c(Br)o1 44211,N1(C(C(C=C)(C)CC)=O)CC(C)(C)C(NC(C2CC=C(C)CC2)=O)C(C)(C)C1 44212,CCC(CC(=O)N1CCC(OCCCNC(=O)CC2CCOC2C)CC1)SC 44213,N1(C(C(C2CCC(C)CC2)CC)=O)CC(CNC(C2CCCSC2)=O)CC1C 44214,C(=O)(CCCC(=O)N(C1CCC(NC(=O)CCCCCOC)CC1)C)NCC 44215,c1(C(=O)NC2C(NC(CC3N(CC)CCC3)=O)C2)c(C)cn(C)c1CC(=O)OC 44216,C(=O)(C1=CCC(C)CC1)NCCC(C)NC(C1(CC(C)C)COC1)=O 44217,C(=O)(CCCCC(F)(F)F)NCC1CN(C(C(CC)C(C)(F)F)=O)CC1(C)C 44218,N1(C(C(CC)(C)C#N)=O)CC2CN(C(=O)C(C)c3ccsc3)CC2C1 44219,CC12CCC(C(=O)NC3CCC(NC(C4(C5CCC5)CCC4)=O)C3)(CO1)C2 44220,N1(C(C2=C(C)CC2)=O)CC2(CC(NC(=O)C(c3ccnn3C)O)CO2)C1 44221,Cc1nccnc1C(=O)N(CC(C)(C)C(=O)NCC(C)(C)CN(C)C)C 44222,C(C)(CCC(=O)N(C)CCN(C(=O)COC(C)(C)C(F)(F)F)C(C)C)SC 44223,CN1CCOCC1c1n[nH]c(CNC(=O)NC(c2ccccc2)c2cccs2)n1 44224,C1(NC(C(CCC)c2ccccc2)=O)CN(C(c2ccc(F)cc2)C)CCC1C 44225,c1(C(=O)OC)cccn(CC(N2CCC2CNC(C2(C(C)C)CCC2)=O)=O)c1=O 44226,N1(C(C(CCSC)(C)C)=O)CCC2(CCCN2C(c2ncc(Cl)cc2Cl)=O)C1 44227,N1(C(c2cc(Cl)nn2C)C(=O)NCC(C)C)CCOC2(CCSC2)C1 44228,C1(C(=O)NC(c2ncc(C)[nH]2)CC)CCN(C(C2CC23CCCC3)=O)CC1C 44229,C(=O)(C#CC(C)(C)O)NCC1CC(COC)CN1C(C1CC2CC1CO2)=O 44230,c1(C(=O)NCCC2(C(=O)NC(C(C)(C)O)CCO)CC2)ccn2cncc2c1 44231,N1(C(C(CC)NC(N)=O)=O)CC2(CCN(C(=O)C=C3CCC(C)C3)CC2)C1 44232,c1(OCC)ncc(C(=O)NC2CCC(NC(C3(C)CCOC3)=O)CC2)cn1 44233,C(=O)(C(F)CC(C)(C)NC(=O)Cc1cnn(C)c1)N(C)CCOCCCN(C)C 44234,c1(C(=O)NC(C)(C)CNC(C2CCC(Cn3ccnc3)O2)=O)cc([N+](=O)[O-])n[nH]1 44235,c1(OC)cc(O)c(CNC2CCC(CC(N3CCC(O)C(C)C3)=O)CC2)c(Br)c1 44236,N1(CC)CCCC(C(=O)NCC2(CNC(=O)CN(C)C3CC3)CC23CCC3)C1 44237,C1(C(N2CCOC(C)(CNC(=O)CSC)C2)=O)(COC)CCCNS1(=O)=O 44238,N1(C(c2cn(CC)nc2)=O)CCCC2(CC(NC(=O)CC3CCCC3C)C2)C1 44239,c1(CC)ccc(CNC(C2CC2CNC(C2(C)CCOC2)=O)=O)cc1 44240,N1(C(C=CCOC)=O)CCC(C(=O)NCC2CN(C)CCO2)C1(C)C 44241,N1(C(c2c(C)c[nH]n2)=O)CC2CCCC2(NC(c2occ3c2CCC3)=O)C1 44242,C1(NC(CCNC(=O)CO)=O)CCN(C(=O)CCc2ccc(F)cc2Cl)CC1F 44243,CC(C)C(C)C(C)CC(=O)NC(C)(C)COCCCNC(c1cnc[nH]1)=O 44244,N1(C(C(CC)(C)C)=O)CC23CCCC2(C1)CN(C(c1cnc(N(C)C)nc1)=O)C3 44245,C(=O)(C(CC)N(C)C(C1(C)C=CCC1)=O)NC1CC(CC)C1 44246,N1(C(c2ccc(CC)cc2)=O)CC2CC(NC(c3snc(C)c3Br)=O)C1C2 44247,Cc1nc2ccc(C(=O)NC(C)CN(C)C(c3cc(C4CC4)ncn3)=O)cn2n1 44248,c1(NC(C(c2cnc(-c3ncccn3)s2)N(C)CC2CC2)=O)ccc(Cl)cc1F 44249,Cc1ccccc1C(=O)N(C1CCCC(N(C(=O)Cc2ccsn2)C)C1)C 44250,C(=O)(CC(O)CCCCC)NCC(CC=C)NC(N1CCN(CC)C(=O)C1=O)=O 44251,c1(OC)cc(N)c(Cl)cc1C(N1CC(N(C)C(C23COCC2C3)=O)C2(CC2)C1)=O 44252,c1(C(N(CC(C)NC(C2(C(F)F)CCC2)=O)CC)=O)cc(C)c(Br)c(C)c1 44253,N1(C(C2C(CC)CCN2C(C2CC(F)(CF)C2)=O)=O)CC(CO)CC(C)C1 44254,Cc1c(C(=O)NC2(C)CC(NC(=O)CC3CCCC(=O)N3)C2)nn2c1CCCC2 44255,c1(C(N2CCCN(C(C=CCOC)=O)CC2)=O)cc2nc(C)cc(C)n2n1 44256,C(C(O)C(=O)N1CC=CC1)NC(=O)CC1CCCO1 44257,c1(C(N2CC(CNC(COCCOC)=O)C(C)(C)C2)=O)cc2cc(Cl)ccn2n1 44258,N1(C(CC2(OCC)CC2)=O)CCC(C(=O)NC(C)Cc2cccs2)C(C)(C)C1 44259,c1(C(=O)NCCCCCN(C(c2c(C)snn2)=O)C(C)C)cncc(N)c1 44260,Cc1cccc(Br)c1-n1cc(CNC(=O)C(=O)N(C)C(C)C)nn1 44261,c1(CCC(=O)NC(C2CCN(C(C3C(=C)C3)=O)C2)(C)C)cn(C)c2ccccc12 44262,c1(NC(C2C(NC(CN3CCC(C)C3)=O)COC2)=O)cncc(C2CC2)c1 44263,O(C=CC(=O)N(CCC(C)NC(=O)CC1CC(C)(C)C1)C)CC 44264,CC(C)C(C(=O)NC1CCCN(C(=O)COC(C)(C)C)C1)c1cccnc1 44265,C(C)(CCC(=O)N(CC(O)CNC(=O)CSc1nncs1)C)NC(C)=O 44266,c1(CC(=O)NC2CCN(c3cc(Cl)c(O)nn3)C2)cn2cc(F)ccc2n1 44267,C1(NC(c2cnc(OC)s2)=O)C2CCN(C(=O)COc3ccsn3)CCC12 44268,c1(C(N(C2CCCN(C(c3cnsn3)=O)CC2)CC)=O)ccc2c(c1)CCNC2=O 44269,N1(C(C(C)NC(C)=O)=O)CC(O)(CN(C(=O)CC2COCC2O)C)C1 44270,c1(NC(C(N2CC(CCO)(NC(C3(CCC=C)COC3)=O)C2)=O)=O)ccc(O)cc1 44271,c1(NC(C(=O)NCC(CC=C)NC(=O)C(C)(C)SC)C)ccc(C(F)(F)F)cn1 44272,N1(C(c2c(CNC(C3(C#N)CC3)=O)occ2)=O)CCC(O)(C(F)F)C1 44273,C1(CC)CCC(C)N(C(=O)CCOCCN(C)C(c2nnc(S)n2C)=O)C1 44274,N1(C(C(C(C)C)NC(N)=O)=O)CC2(CNC(=O)C=Cc3ccncn3)CC1CO2 44275,C1(C(=O)NCCC#C)CCN(C(=O)c2cccc(Cl)c2)O1 44276,CC1COc2c(C(=O)NC3C4CC3N(C(c3cc(=O)cc(Cl)[nH]3)=O)C4)cccc21 44277,C1(C)(C(=O)NC(CCC)CO)CN(C(=O)CC2(C)CCC2)CC1C 44278,c1(C(N2CCCC(NC(C3(COC)CC=CC3)=O)C2)=O)cc(C)c(C)nc1C 44279,Cc1nc2[nH]c(C(N3CCC4(NC(c5ccc(F)cn5)=O)CC4C3)=O)cc2s1 44280,C1(NC(c2cn(CC=C)nc2)=O)CC2CCC1CC2NC(C1(C)CC=CCC1)=O 44281,CC1(C(=O)NCCC2CCN(C(=O)COC3CCC3)C2)CCOC1 44282,Cc1nc2cccc(C(=O)N(C(C)CNC(=O)C(F)n3cccn3)C)c2s1 44283,C12(C(=O)NCC(C)N(C(C3(c4cccc(C)c4)CCC3)=O)C)CCC(F)(CC1)C2 44284,C1(CN(C(C(C)C)=O)C)CN(C(C2CCS2(=O)=O)=O)CCO1 44285,c1(NC(C(c2ccccc2F)NC(C(C)=O)=O)=O)cccc2cncc(C)c12 44286,CCCCCC(CC)C(=O)NCC1(CNC(=O)C(n2nccc2C)C)CCCC1 44287,Cc1cc(CC(=O)N(C2CCCC2)CCNC(=O)C(C)(C)ON)n(C)n1 44288,c1(CC(=O)NCCN(C(=O)C(C)(O)CC)CC)ccccc1S(=O)(=O)C(F)F 44289,C(C(=O)NC12CC(CNC(=O)CSC(F)F)(C1)C2)(c1ccccc1)=C(C)C 44290,Nc1cccc(F)c1C(=O)NCC1CCN1C(=O)C(c1ccncc1)C1CCCO1 44291,C(=O)(CCCC(C)(C)C)N1CC(CC)C(NC(c2cccc(OC(C)C)c2)=O)C1 44292,CC(C(C)N(CCCC(=O)NC1CC1)C(=O)CN)S(C)(=O)=O 44293,c1(OC)cc(Cl)ccc1CNC1CC1C(N1CCC2(CC1)CC2)=O 44294,C1(NC(N(C2(CN(C)C(C3CSCCS3)=O)CC2)C)=O)CCCC1c1nc[nH]n1 44295,N1(C(C(C(C)(C)C)N2CCCC2)=O)CCC2(CC1)CC2CNC(c1ccon1)=O 44296,C1(C(=O)NC2C(CNC(=O)CCC3CCCCO3)CCC2)CC2OC1C1CC21 44297,C(=O)(C1COc2ccc(Cl)cc21)NCCN(CCC)C(C1CCC1C(F)(F)F)=O 44298,N1(C(CCC=C)=O)CCC2(CCCCN(C(=O)C(C)N(C)C)C2)C1 44299,C1(CC)CN(C(c2ncc(Br)cn2)=O)CCC1NC(=O)C=CC(C)(C)C 44300,c1(CNC(C2(C)CN(C(=O)CC3CC4CCC3C4)C2)=O)cnc(C(F)F)nc1 44301,n1(CC)cc(Cl)c(C(=O)N(C(C)CCNC(=O)Cc2ncc(C)s2)C)n1 44302,N1(C(c2cnc(CC(C)C)s2)=O)CCCC(C)(NC(c2cc(F)cc(Cl)c2)=O)C1 44303,c1(OC)cncc(C(=O)NCC2CN(C(=O)CSCc3cccs3)CC2O)n1 44304,c1(C(=O)NCC2N(C(C34CCC(C)(CC3)CC4)=O)CC2)cccc2c1COCC2 44305,C(C(C)C)(C(O)C(=O)NCC(c1ccccn1)C)OC 44306,N1(C(C2CCCN(CC)C2)=O)CCCC2CN(C(=O)C(F)CC3CCCC3)CC12 44307,c1(C(N2CC(CNC(C3(CCCC)CCC3)=O)C(C)C2)=O)cc2c([nH]1)CCCC2 44308,O(N(C)C(=O)CN=c1[nH]c(=NC(C)CC2CCCO2)[nH]c2c1COCC2)CC 44309,C=CCCCC(C(=O)NC1CCC(C(N)=O)C1)NC(=O)CC1(OC)CCC1 44310,[N-]=[N+]=NCCCCCCC(=O)NCC1CN(C(=O)CC23CCCC2C3)C1 44311,C1(C)(C(=O)NCC(C(C)C)(C)NC(c2nn(C)cc2Cl)=O)CCCCCC1 44312,c1(OC)ccc2cc(C(N3CC(NC(C4CCC(F)CC4)=O)C3)=O)[nH]c2c1 44313,c1(NC(C2CCN(Cc3ccc(C)[nH]3)CC2O)=O)cccc2c1OCO2 44314,c1(N(C(C(n2c(CCCC)ncc2)C)=O)CC2CC2)ccc(F)cc1 44315,C(=O)(C1=C(Cl)CCCC1)NC1CN(C(Cc2c(C)scc2)=O)CC(F)C1 44316,C1(CNC(C(C(=O)OC)(C)C)=O)CCN(C)C1=O.C123CC(C1)(C2)NC3=O 44317,Cc1sc(Br)cc1S(=O)(=O)N1CCC2(O)CCOCC2C1 44318,S(=O)(=O)(c1ccccc1)N(CCN(C)C(=O)Nc1cc(O)cc(F)c1)C 44319,N1(C(CCS(=O)(=O)NC)=O)CC2CC1CCC2NC(C1CCCC(C(=O)OC)C1)=O 44320,N1(C(CC(c2ccc(C)cc2)C)=O)CC2CC(NC(=O)CC3CC=CCC3)C2C1 44321,c1(CC(C(N)=O)NC(C2CCCN2C(c2ncccc2F)=O)=O)ccc(O)cc1 44322,CN1CCOCC1CC(=O)NCc1ocnc1Cn1cc(C2CC(F)(F)C2)nn1 44323,C12(COC)COC(C(=O)NC3CCCCC3NC(c3c(C)coc3SC)=O)(C1)C2 44324,Cc1ccc(C)c(C(N2CC3C(CNC(=O)CC(C)O)C3C2)=O)c1 44325,C1(NC(C2CCC(C)O2)=O)COCCN(C(c2cccc(Br)c2F)=O)C1 44326,N1(C(C(SC)SC)=O)CC(NC(=O)Cc2cc(C)on2)CC(C)C1 44327,C#CCC(C)(C)CNC(=O)C(CCOC)NC(c1[nH]ccc1C)=O 44328,c1(OCC(=O)NCCC2CCCN2C(=O)CC2COCC2O)ccc(F)cc1 44329,N1(C(C(N2CCSCC2)C)=O)CC2CCN(C(c3cccc(N)c3)=O)C2C1 44330,C1(C(=O)NCC2CC(NC(c3cnc(C(C)=O)s3)=O)C2)Cc2ccncc2C1 44331,C(=O)(CC(C)CF)N(CCOCCOCC#C)CC.C1C(=O)NCCCO1 44332,C(=O)(N=c1c(Br)c[nH]cc1I)C1CCC(NC(c2ccc(F)c(F)c2Br)=O)CC1 44333,C(N=c1[nH]c(=NCCC=CBr)[nH]c2c1CCCCCC2)C1(C)CCC(=O)N1 44334,c1(CNC(=O)CC2(O)CN(C(c3c[nH]nc3C3CCCO3)=O)C2)ccccc1 44335,N1(C(c2cc(C)no2)=O)CCC2CCC(C1)N2CC1CCC2CC2C1 44336,O=C1CCc2c(C(N3CCOC(C4CC(F)(F)C4)C3)=O)n[nH]c2C1 44337,c1(C(=O)O)ccnn1Cc1cn(CC(N2CCC(N3CCCC3=O)C2)=O)nn1 44338,C1(C(C)NC(Cn2ccc(C)n2)=O)CCCCN1C(=O)CNC=O 44339,C1(CN(C)C(C2CC23CCC3)=O)CCN(C(c2ccccc2OCC#N)=O)CC1 44340,C1(NC(C(C)C2CCC2)=O)CN(C(c2cc3cnccc3[nH]2)=O)CC2CCCC12 44341,C(=O)(C(CCC1CCC1)NC(c1c[nH]c(=S)cn1)=O)NC(CCC)COC 44342,C1(NC(c2ccn3nccc3c2)=O)CN(C(=O)CC2(O)CCOC2)CC2(CC2)C1 44343,C(=O)(CC1(O)CCOc2ccccc21)N1CC(C)(C)c2c1cccc2 44344,c1(CCC)cc(C(N2CCC(C(C)CNC(C3(CO)COC3)=O)CC2)=O)n(C)n1 44345,c1(OC)cc(C)c(C(N2CC=CC(NC(=O)Cc3ccn(C)n3)C2)=O)cc1Cl 44346,N1(C(C2(NC(C(CC=C)OC)=O)CCC2)=O)CCN(C2CC2)C(C)C1 44347,N1(C(c2c(C)cccc2)=O)CC2CCCC(C1)N2C(=O)COC1CCCCC1 44348,c1(C(=O)NCC(CCCC)NC(=O)C(CC(C)C)OC)cc(OC)cc(C)c1N 44349,N1(C(CC2(NC(c3cc(CC4CC4)on3)=O)CC2)=O)CC(O)(C(F)F)C1 44350,N1(C(C(c2cn(CC)nc2)=O)=O)CCN(C(=O)CCC(C)OC)CC1CCOC 44351,C(C(=O)NN1CCC(c2cn[nH]c2)CC1)(C(C)(C)C)NC(=O)OC(C)(C)C 44352,c1(C(=O)NCC2OCC(CNC(=O)C(Cl)=CCl)C2)cnn2ncccc12 44353,N#CC1CCCC(C(=O)NC2CC(CNC(=O)COc3cc(F)cc(F)c3)C2)C1 44354,C12(NC(C3C4CCN(C(=O)CN5CCCC5=O)CC43)=O)CCC(O)(CC1)CC2 44355,c1(C(N2CCCCC(NC(C(CC)(C)OC)=O)CC2)=O)c(F)cc(C#N)cc1F 44356,C1(C(=O)Nc2cnc(C)s2)CC(C)CN1C(=O)C(=O)Cc1ccc(O)cc1 44357,C1(CNC(c2cc(OC)ncn2)=O)CCC2(CO1)CC(NC(c1cncs1)=O)C2 44358,c1(C(=O)NCC2(CNC(CCCOC)=O)CC23CCC3)cc(OC)cc(C#N)c1 44359,Cc1ccc(NCC2CCN(c3ccc(F)cc3F)C2)cc1Br 44360,CN1CCN(C(=O)CC2(O)CCCCC2)CC1CNC(=O)Cc1cncnc1 44361,Nc1cc([N+](=O)[O-])ccc1C(N1CC(NC(=O)Cn2cccn2)C2(CCC2)C1)=O 44362,c1(C(=O)NCC(C)(C2CCC2)NC(C2CC2F)=O)cc(Cc2ccccc2)c[nH]1 44363,C(C(=O)NC(CCSC)C(=O)NCC1C=CCC1)(C(C)C)OCC 44364,c1(OC(c2nc(-c3nccs3)nn2C(=O)NC2CC2)C)ccc(F)c(Cl)c1 44365,C=CCN=c1[nH]cc(C(=O)NC2COCCN(C(C3CCCCC3(C)C)=O)C2)s1 44366,C=C1CC2CCCC(C1)N2C(C1CC(NC(c2ccc(C)cc2F)=O)CCO1)=O 44367,N1(C(C23CC(C)C2C3)=O)CCC2(CC1)CC2CNC(c1cnn(C)c1Cl)=O 44368,c1(NCC(N)=O)[nH]c(=NCC2CC=CCC2)nc2scnc12 44369,Cc1ccc(N2CCOC(C(=O)NCC3CCN3C(=O)OC(C)(C)C)C2)nc1Br 44370,C#CCC(C)(CC)C(=O)N1CCC(c2cccc(F)c2)(NC(=O)CC(F)F)C1 44371,c1(CC2CCCN(C(N3CC(N(S(C)(=O)=O)C)C3)=O)C2)cccnc1N 44372,CCC(C)(COC)C(=O)NC(CNC(=O)C1=COCCC1)C1CCC1 44373,C12(CC)CN(C(=O)Cn3cnnn3)C(CNC(C3CCS(=O)(=O)N3)=O)(C1)C2 44374,N1(C(C(C)OCCC(C)C)=O)CCC(O)C(NC(=O)CN2CCC(C)(C)C2)C1 44375,c1(-c2cn(CC3N(C(CC(COC)O)=O)CC=C3)nn2)cccc(C)c1Br 44376,O=C(C1=CCC(F)(F)CC1)N1CCN(C(C2(C3CCCO3)CC2)=O)C(CCO)C1 44377,N1(C(CCC2CCN(C(C(C)C3CCCO3)=O)CC2)=O)CCc2n[nH]cc2C1 44378,CC1CN(C(c2csc([N+](=O)[O-])c2)=O)CCCN1C(C1CC(=O)NC(=O)C1)=O 44379,C1(CC)CN(C(CCC2CCC2)C(=O)NCc2ccco2)CC1O 44380,C(C(=O)NCC(O)CCNC(=O)CCCc1cccnc1)(C(C)O)NC(C)=O 44381,c1(C(=O)NC2(C(N(CCCF)CC)=O)CC2(C)C)cnn(C)c1C#N 44382,C(=O)(CC(C)(C)CN(C)C)NC(C(C)C)CNC(=O)C(C)C1CCCC1 44383,CC1(C)C(CC(=O)NCCCCCO)CCN1C(=O)C(O)CN1CCCC1 44384,Cc1nc(C(N2CC(NC(c3ncccc3Br)=O)C(O)C2)=O)n(C)n1 44385,CCC(C(=O)NC(C(=O)NCCC1CCCCO1)C1(C)CC1)N(C)CC 44386,C(=O)(C(F)(F)C(C)(C)O)N1CC(NC(C(CSC)C)=O)C(C(F)(F)F)CC1 44387,C1(Cc2ccccc2)CC(=O)N(C(=O)OC2CC2)C1.C1(CC)CC(OC)C1 44388,CCC(C)CCC(=O)N1CCCC1CCC1CCN(C(C2CC2C(C)C)=O)CC1 44389,Cc1cc(=NC2CC(NC(c3c[nH]cc(F)c3=O)=O)C2(C)C)[nH]cc1C#N 44390,C1(NC(c2ncc(C)c(C)c2)=O)CN(c2nnco2)C2CCCCC12 44391,C(=O)(CCCCC(N)=O)N1CCC(=C)CC1C(=O)NOCC1CC2C=CC1C2 44392,C(=O)(C#CC1CCCOC1)NC1CC2CN(C(c3cc(C#N)sc3)=O)CC21 44393,C1(NC(C2C(CCOC)C2)=O)COCCC1NC(c1nc(OC)c(C)s1)=O 44394,C(C1c2ccsc2CCN1C(c1[nH]ncc1C#N)=O)NC(C(CC(C)C)OC)=O 44395,N1(C(c2cn(CCC)nn2)=O)CCN(C(=O)CC(CC)C(C)C)CC2(CC2)C1 44396,CC(C)C(C(=O)N1CCC(CCNC(C2CC2c2cccnc2)=O)CC1)N(C)C 44397,C1(C(N2CC(C(N3CC(C(=O)NC)OCC3)=O)OCC2)=O)CCOC(=O)CC1 44398,c1(C(N2CCC(CSc3ccccc3)C2)C(=O)NCC)ccn2nccc2c1 44399,c1(C(CC)NC(N2CCCC(N3CCNC3=O)C2)=O)ccc(Cl)c(F)c1 44400,C#CC1(C(=O)NCC2CC2Cl)CN(C(=O)CC2CCCC2C)C1 44401,O=C(C1=CCCN(C(c2cc(Cl)ncc2F)=O)C1)Nc1ccc(OC(F)F)cn1 44402,CC1CC(NC(=O)C(F)=CC2CC2)CN(C(=O)C(C)(O)c2ccccc2)C1 44403,c1(C(=O)NCC(C)CNC(=O)C(C)C2CC2)ns[nH]c1=O 44404,c1(OC)ccc(CC(=O)N(CC(C)NC(=O)Cc2c[nH]ccc2=O)C)c(C)c1 44405,N1(C(c2cnc(C)s2)=O)CC(N=c2[nH]c3c(C)cccc3o2)C2(CCC2)C1 44406,C(=O)(CN=c1cc[nH]cc1)N1CC(NC(c2occ3c2CCC3)=O)C2C1CCC2 44407,C1(CNC(C(CC)F)=O)CC2(CCN(C(=O)CCc3cc(Cl)no3)CC2)C1 44408,c1(C(=O)NCC(c2ccsc2)O)cc2cccc(Br)c2o1 44409,N1(C(C2(C(CC)=O)CC2)=O)CCN(CC(=O)NCC2CCN(C(C)=O)C2)CC1 44410,C1(NC(c2c(C)[nH]nc2C(F)(F)F)=O)CN(C(c2cncnc2)=O)CCC1CO 44411,C(C1=NOC2(COC2)C1)N1C(=O)CN(c2ccc(Br)c(F)c2)C1=O 44412,c1(OC)ccc(CNc2ncnc(NCCC(O)COC)c2C)c(OC(F)F)c1 44413,c1(C(N2CC(C)(NC(CCC(CC)C)=O)C2)=O)nc(O)nc(O)c1N 44414,c1(C(N(C(CCNC(c2c(Cl)cn(CC)n2)=O)C)C)=O)ccc2cnccc2n1 44415,CC1=NNC(=O)C1CC(N1CCOC(CCNC(=O)C(C)(C)C2CC2)C1)=O 44416,C1(CC(=O)NC(CC)(C)CNC(c2cn[nH]c2)=O)Cc2cccc(Cl)c2O1 44417,C1(NC(COCCOCCOC)=O)CN(C(=O)Cc2ccno2)C2(CCOC2)C1 44418,CCCC(O)C(CO)NC(=O)NC(Cc1ccccn1)CO 44419,c1(CC)ccc(OC)cc1C(N1CCCC1C(C)NC(C1(Cl)CC1)=O)=O 44420,C1(CNC(C2C(CCC)C2)=O)CCC(CNC(C2CCC3(CC3)C2)=O)CC1 44421,C12(NC(C3CC(=C)C3)=O)CCC(CC1)N(C(=O)C(C)(C)NC(=O)OC(C)(C)C)C2 44422,C(CC1c2ccccc2CCN1C(=O)C(C)C(C)C)NC(CCOCCOC)=O 44423,C12(C(N3CCCC(CNC(Cc4ccc(OC)cc4)=O)C3)=O)CCC(C)(C1)OC2 44424,c1(NC(CCC=C)C)[nH]c(=NCCc2noc(=O)n2C)nc2ncn(C)c12 44425,N1(c2ncc(C)c(O)n2)CCC2(CC1)OCCCC2NC(C1CC1(Cl)Cl)=O 44426,C=C(C)c1ccccc1NC(=O)CCOC1CN(C(C2OC3CCC2C3)=O)C1 44427,C1(NC(CC(CNC(=O)CC2(O)CCOCC2)OC)=O)CCn2cncc2C1 44428,C1(C(N(C)C)=O)CCCN(C(=O)C(=O)NC2COCC2OC2CC2)C1 44429,c1(C(=O)NCC2CC(COC)CN2C(C2CC(C)(F)C2)=O)cc2cccnc2s1 44430,CC1(CNC(=O)CCN2CCOCC2)CCCN1C(=O)CC1(CO)CC1 44431,C1(CN(C(CC2C(CC)C2)=O)C)CN(C(c2ocnc2C)=O)CC12CC2 44432,c1(SC)cc(=NC(=O)C2CCN(C(=O)CC3CC=CCC3)CC2C)[nH]n1C 44433,c1(CC(=O)NCCCCNC(C=CC(CC)C)=O)ccc(Cl)c(F)c1 44434,c1(OC)c(C(=O)Nc2cncc(-c3ccc(SC)cc3C)c2)ccc(Cl)c1Cl 44435,c1(C(=O)NC2C(C)N(C(=O)CC3CCCCN3C)CC2)cc(F)cc2ccoc12 44436,C=CCC(C)(C)CC(=O)N1CCN(C(=O)Cc2cc(OC)no2)CC1CF 44437,C12(C(=O)NC(c3c(C)cccc3)C)CC(C)(CN1C(c1cc(O)n(C)n1)=O)C2 44438,c1(NC(C(C)C)CNC(=O)CC2CCCOC2)ncncc1I 44439,c1(CN(C(c2csc(C)n2)C(=O)NCCOCC)C)cccc2c1OC(F)(F)O2 44440,N1(C(C(=O)Nc2cccc(C(C)(C)C(F)(F)F)c2)=O)CC(CO)CC(C(=O)O)C1 44441,C1(CCNC(C2(C=C)CC2)=O)CN(C(C2OCCC2C(F)(F)F)=O)CCS1(=O)=O 44442,C1(C)(CNC(C2(CCCC)CC2)=O)CCN1C(=O)OC(C)(C)C 44443,Cc1cc(C(=O)N(CC(=O)N(C)C(C2CCCCC2)C)C2CC2)cc(C)n1 44444,C(C(O)C(=O)N1CCC1c1cn(Cc2occc2C(=O)O)nn1)OC 44445,Cc1cc(C)c(C(=O)NCC2CCN2C(=O)CSc2ccc(CO)cc2)c(S)n1 44446,C1(NC(C(COC)(F)F)=O)CCC(C)N(C(c2ccc(-c3ccco3)[nH]2)=O)C1 44447,O(NC(=O)C(COC)NC(C12CC1CNC2=O)=O)CCOCC#C 44448,N1(C(C(CC#C)C2CC2)=O)CC(C)(C(=O)NC2(C3CCCO3)CC2)CC1(C)C 44449,c1(NC(C2C(C(=O)Nc3ccc4sncc4c3)C2)=O)c(O)cccc1[N+](=O)[O-] 44450,N1(C(CCCNC(C)=O)=O)CCN(C(=O)C(c2ccc(Br)cc2)C)C(C)C1 44451,n1(CC=C)nnnc1C(c1ccc(-c2ccccn2)s1)NCc1ccc(CC)o1 44452,CCC(C(=O)N1CC(CNC(=O)CCN(C)C(C)C)C1)c1ccccc1 44453,C=CCC(CNC(C1C2CCC(C2)C1C)=O)C(=O)NC1CCN(C(=O)CC)C1 44454,C1(c2cn(CC(C)NC(=O)CSC(F)(F)F)nn2)COC(C)(C)O1 44455,C1(NC(c2ccc(O)nn2)=O)(CO)CCCN(C(=O)Cc2ccc(O)cn2)C1 44456,C(C(C)CC(=O)NCCC1(OC)CN(C(C2COCCN2C)=O)C1)OC 44457,c1(CC)oc(C(N2CC(CC(=O)NCC(C)CC3CC3)C(C)C2)=O)cc1C 44458,n1(C2CN(C(=O)Nc3c(C)oc(SC(C)C)n3)C2)ccc(O)nc1=O 44459,C1(C(N2CCOCC2)C)CCCCN(c2nc(=N)nc(N3CCC(N)C3)[nH]2)C1 44460,C1(NC(c2cc(C)ncn2)=O)CC2(C1)CC(C(=O)N(CC(N)=O)C)C2 44461,C(=O)(C1=CCCC1C)NCC1CC(COC)CN1C(c1ccccc1)=O 44462,C1(C(C)C)(C(=O)NCCC2CN(C(=O)C(O)C(F)F)C2)CNC(=O)C1 44463,c1(OC)ccc(NC(C2CC3CC3N2C(=O)Cc2ccccc2OC)=O)cc1C 44464,C(CCN(C)C)(C(=O)N1CCOCC1CCO)NC(c1scc(C)c1)=O 44465,c1(N(CCNC(c2ccc(-c3cc[nH]n3)s2)=O)CC2CC2)nc(O)n[nH]1 44466,c1(C(=O)NC(C2CC2C(=O)NCCC2CC2C)C)cnnn1C 44467,N1(C(C2(C#C)CC(=O)C2)=O)CCC2(CC1)CN(C(c1cc(C)n(CC)n1)=O)C2 44468,C(C(=O)N1CCC(F)(C(=O)NCC2CC(N(C)C)C2)C1)(C(C)(C)C)OC 44469,S(=O)(=O)(c1ccc(F)cc1)NC(CC(=O)N(CC(C)NC(C1(O)CC1)=O)CC)C 44470,C1(COC)(CNC(=O)CC2CC(OC)C2)CCN(C(C2OCCC2C)=O)C1 44471,N1(C(C2(CC)CCCN2C(C2CCC(N(C)C)C2)=O)=O)CC(C)OC2(CCC2)C1 44472,C(=O)(C(CNC(=O)CCn1cnnc1)C(C)(C)C)NCc1cn(CC)nn1 44473,N1(C(C(c2c(C)cncc2)C)=O)CC2(C1)SCCC2NC(=O)CSc1cn[nH]c1 44474,N1(C(COC(C)C)=O)CCC(C=CC(=O)NCC2CC(C)CO2)CC1 44475,N1(C(CNC(=O)OCC=C)=O)CCC2(CC1)CC2NC(C1CC12CCC2)=O 44476,c1(C(=O)NC(C2N(C(C(CC3CC3)OC)=O)CCC2)C)ncc(Cl)cc1F 44477,C(=O)(CC(C)P(C)(C)=O)NCC(CCCC)NC(c1cc(OC)n(C)n1)=O 44478,Cc1cc(Cl)c(C(=O)NCC2(F)CCN(C(c3cnncc3O)=O)CC2)cc1C 44479,n1(CC(N2C3CC(CNC(C(C)OC)=O)CC2CC3)=O)cnc2cc(C)ccc12 44480,C1(C(=O)NCCC(C)Nc2cncc(C#N)n2)CCc2nn[nH]c2C1 44481,c1(C(N(C)CC2CCCN2C(=O)C(=O)NC2CC2)=O)ccc2c(c1)CCCCN2 44482,n1(CC(=O)NC2(CO)CN(C(=O)CCC3CC3(F)F)C2)nnc(C2CC2)n1 44483,CCCC(CC)C(=O)NC1(CC)CCCN(C(c2ccoc2)=O)C1 44484,c1(C(N2CC(=C(CNC(CCNS(CC)(=O)=O)=O)F)C2)=O)cc(C)ccc1F 44485,CCC(CCO)N=c1[nH]c(N2CCCC(COc3ncccc3Cl)C2)nc(=N)[nH]1 44486,CC1(NC(=O)C(C2CCN(C(=O)Cc3csnn3)C2)F)CC2(CCC2)C1 44487,C12(CCNC(c3c(C)noc3)=O)CCC(CC1)N(C(c1ccc(F)c(F)c1)=O)C2 44488,c1(COC)ccccc1C(=O)NC(C)C(C)NC(c1cc(Br)cn1C)=O 44489,Cc1cc(F)c(CNC2CN(C(c3cc(Br)nc(Br)c3)=O)CCC2(F)F)cc1Br 44490,Cc1c(C(=O)NCC2(NC(C3CC(=O)CCO3)=O)CCC2)cncc1F 44491,c1(OC)cnc(C(=O)NCC(C)(C)OCC(=O)NCC(N)=O)cn1 44492,c1(C(N2C(CCNC(C(C)OCCCC)=O)CCCC2)=O)cc(F)c(C)cc1Cl 44493,CC1CCN(C(C2COC3(C2)CN(C(=O)C(F)Cl)C3)=O)CCC1O 44494,c1(CCC(=O)N(C)CC2N(C(CC(C)F)=O)CCOC2)nnc(S)nc1O 44495,C1(CC(=O)O)CC2(CCOCC2)CN1Cc1cc(N)c(O)c(F)c1 44496,c1(C(N2CC(CC(C)C)C2)=O)cc(CNC(c2cnco2)=O)on1 44497,c1(N2CC3CN(C(CCCC=C)=O)CC32)ncnc2ccc(OC)cc12 44498,C1(C(=O)NCC2C(CC(=O)NCCN3CCC(OC)C3)C2)(CF)CNC(=O)C1 44499,C1(NC(=O)NCc2ccc(OCCCCOC)cc2)CCC2OCCC2C1 44500,N1(C(C#CC)=O)CCc2[nH]nc(NC(=O)CCN3CCOCC3)c2C1 44501,c1(C(=O)NC2CN(C(c3cc(SC)oc3)=O)C(C)CC2)ccc(P(C)(C)=O)cc1 44502,N1(C(c2cc(OC)ncc2)=O)CC(NC(=O)C(=C2CCCCC2)F)C(N=[N+]=[N-])C1 44503,c1(C(=O)NCC2C(NC(C(C)SC(C)C)=O)C2)cc(C(F)(F)F)ncc1Cl 44504,C12(NC(=O)CC(F)(F)Cl)CCC1CN(C(c1ccc(-c3cccs3)o1)=O)C2 44505,N1(C(c2c(CC)csc2)=O)CC2CC(C(=O)NCCN3CCOC3=O)CC2C1 44506,c1(OCC(=C)C)ccccc1COC(C1(CF)CCNCC1)=O 44507,CC1CCCC(N(C)C(C2CC3(CC(NC(=O)Cn4ccnn4)C3)C2)=O)C1C 44508,C(c1cc(C)n(CC)c1C)=C(C(C(=O)OCCC)NC(=O)C(CC(C)C)OC)C 44509,C1(OC)CN(C(=NCCc2sccc2C)NCc2ccco2)CC1O 44510,C1(C(=O)NCCCNC(C(C)C)=O)CC(C)N1C(=O)C=Cc1ccoc1 44511,O=S(=O)(c1cccc2cccnc12)NC1C2CCC1CN(Cc1cnc[nH]1)C2 44512,c1(CN(C(c2ccc(C)o2)C(=O)Nc2cn(C)cn2)CCCC)ccc(F)cc1 44513,N1(C(C(CC)N(C)C)=O)CC2C(NC(=O)CCc3cccnc3)CS(=O)(=O)C2C1 44514,C1(CC)(NC(=O)CC2CCCO2)CCN(C(=O)C=CSc2ccccc2)CC1 44515,c1(C(=O)OC)ccc(O)nc1NC(C)CC(C)NC(C1CCS(=O)(=O)C1)=O 44516,c1(NC(CNC(c2ccc(COC)s2)=O)C)ncc(Br)cc1C#N 44517,c1(CC(N2CCC(N(C(=O)CCCc3ccccn3)CC)C2)=O)c(C)n[nH]c1C 44518,C1(C(=O)NC(C(C)NC(c2ccnnc2)=O)CO)CCCC2(CCCCC2)C1 44519,c1(NC(=O)Nc2c(C)cc(Br)cc2F)c(C#N)oc2ccccc12 44520,N1(C(c2cc(C)n(C)c2C)=O)CCC(NC(=O)CCC2CC2(C)C)CC(C)(C)C1 44521,N1(C(c2cccc(C(C)=O)c2)=O)CCC(NC(C2CC3C=CC2C3)=O)C(C)(C)C1 44522,C1(C(=O)NCc2ncco2)(CC)CCCN1C(=O)CCN(C)C 44523,N1(C(CCC(=O)NCCC)=O)CC2CCCN(C(=O)C=CCOC)C2C1 44524,C1(CC(=O)NC2(CO)CN(C(=O)CC3CCS(=O)(=O)C3)C2)CCCC1(F)F 44525,Cc1cnc2ccc(C(=O)NC3CCN(C(=O)CCS(C)(=O)=O)C3)cn12 44526,S(=O)(=O)(c1cnn(C2CC2)c1)N1C(C(N2CCCC(C(=O)O)C2)=O)CC2CC21 44527,Cc1ncncc1C(N1CCC(N2CCN(C(C3CCCCN3C)=O)CC2)C1)=O 44528,c1(C(N2CC(CNC(CN3CC(CC)C3)=O)OCC2)=O)cccc2ncc(C)n12 44529,N1(C(CC2CCC(=O)C2)=O)CC2(CCCC2NC(c2cccc(C3CC3)c2)=O)C1 44530,c1(C(=O)NCCCC(C)NC(c2ncc(OCC)nc2)=O)c[nH]c2nccc-2c1 44531,C1(CNC(C(CCC)OC)=O)CC2(CO1)CN(C(=O)CC(F)(F)C(C)C)C2 44532,c1(C(=O)NCCN(C(=O)CC2=CCCC2)CC(C)O)cc2n(c(=O)c1)CCS2 44533,C12(C(=O)OC)CC(NC(=O)NCCC(N)=O)CC1C2.c12ccc(cc1)CN2C 44534,c1(CC)ncnc(CC)c1C(=O)NCCN(C(=O)C(O)CC(N)=O)C 44535,CC(C(=O)N(C(C)C(F)F)C)C(C)NC(=O)C=Cc1cscn1 44536,N1(C(C(c2ccc(F)cc2)OC)=O)C2CC1CN(C(c1cnc(C3CC3)[nH]1)=O)C2 44537,C1(C)(CC)CCN(C(C2CC2C2CN(C(C3(C)CCCN3C)=O)C2)=O)CC1 44538,N1(c2nc(CC)nc(=N)[nH]2)C2CCCC1CN(C(=O)C=C1CCCC1)C2 44539,c1(C(C(=O)NCC(CNC(c2cc(Cl)ccn2)=O)OC)=O)ccc(Cl)cc1 44540,Cc1cnn(CC(N2CCC3C(NC(=O)CN(C(=O)C(C)C)C)C3C2)=O)c(=O)c1 44541,c1(C(=O)NCC2CCN(C(c3c(C)nn(C)c3C)=O)C2)cnn2cccc(C)c12 44542,c1(C(=O)NCC2(CNC(=O)CC(F)F)CCCC2)ccc(O)cc1F 44543,C(C)(C(=O)N(CCCN(C)C)CC)NC(CC)=O.C12CC(C1)CC(=O)NC2 44544,c1(CC(C)C)cc(C(N2CCC(CNC(=O)CC3(C)CC3F)CC2)=O)cc(O)n1 44545,C1(NC(c2cnc(Cl)n2C)=O)CCC(C)(C)C1.C12CC(C1)C(=O)N2C 44546,N1(C(COCP(C)(C)=O)=O)CCCCC(NC(c2ccc(N3CCC3)nc2)=O)C1 44547,Cc1ncn(C)c(=O)c1C(=O)NCC1C(C)CCN1C(=O)C(F)=C1CCC1 44548,C1(CNC(c2csc(C(F)F)n2)=O)(CO)CCN(C(C2CC3(CC3)CO2)=O)C1 44549,c1(C(N2C(C)(CC(=O)N(C3CCOC3)C)CC2)=O)cnc(=N)[nH]c1 44550,CCC(C)C(C(=O)NOCc1nc[nH]n1)NC(c1ncc(F)cc1N)=O 44551,C1(C(=O)NCC)(NC(=O)C(COC)NC(=O)CC(=O)N(C)C)CCCC1 44552,C12(SCC)CC(NC(=O)N)(CO1)C2.C1(C)(C2CC2)CC(C(=O)NC)C1.C1(=O)CN1 44553,C1(C(=O)NCC2CC(NC(=O)CC3CCCC34CC4)C2)CC2(C1)CC1(CC1)C2 44554,N1(c2n(CCOCCC=C)c(-c3cn(C)nn3)nn2)CC(C)C(F)(F)C1 44555,c1(C(=O)NCC2CC(CC)C2)cc(CNC(c2cccnc2O)=O)ccn1 44556,Cc1cncc(C(=O)N(C)CCOCCCNC(C2CCC(N(C)C)CC2)=O)c1 44557,C(CN=c1cc(NCc2n[nH]cc2C)nc[nH]1)(C1CC1)OC 44558,c1(C(=O)OC)ccnc(C(N2CCC(O)(CN(C)C)C2)=O)c1.C12(CC1)CNC2 44559,C1(C(N(CCN(C)C(c2cccnc2)=O)C)=O)CCCC2CCCN12 44560,c1(C(=O)NCCC2N(C(CC3CCN(C)C3)=O)CCC2)cn(C)ccc1=O 44561,N1(C(C(COC)(F)F)=O)CCC(C2(O)CN(C(C3CCCS(=O)(=O)C3)=O)C2)CC1 44562,CC1CN(C(=O)CCc2cn(C)cn2)CCN(C(=O)C(O)C(F)(F)F)C1 44563,c1(CN(C)CC2CCCN2C(C2CC3CC2C2CC32)=O)ccc2nonc2c1 44564,C1(NC(c2cnn(CCC)c2C)=O)CC(C)CN(C(=O)CC2CCCC2(F)F)C1 44565,N1(C(C2(CC)CC2)=O)CCC2(CC1)CC2NC(=O)C(c1cc(C)cc(F)c1)C 44566,c1(SCC)ccc(Cl)cc1C(=O)NCCCN(C(C1(O)CCCC1)=O)CC 44567,C(=O)(CCS(=O)(=O)CC(C)C)N1CCCC(O)(CNC(C(CCC)OCC)=O)C1 44568,Cc1cccc(C(N2CCC(CN(C)C(C3CCS(=O)(=O)C3)=O)C2)=O)c1Cl 44569,c1(C(N2C(C(=O)O)CC(NCCCCS(C)=O)C2)=O)cccc2c1OCCO2 44570,C1(C(=O)NCCN(C(CC(=O)OC)=O)C2CCCC2)CC(O)C(F)C1 44571,c1(C(=O)NCc2c(CC)noc2C)coc2c1CN(C(c1ccc(C)n1C)=O)C2 44572,C1(C(C(=O)NCC2CCN2C(c2cnc(C)cn2)=O)OC)CCC(F)(F)CC1 44573,N1(C(c2cccc(OC)n2)=O)CCc2ccc(C(=O)NCCCC(C)C)nc2C1 44574,CCC(CC)CCCC(=O)N1CC2CC2(NC(=O)Cc2nc(F)c(F)cc2F)C1 44575,c1(NC(CN(C)C)C(=O)N2CC(c3ccccc3F)(C)C2)cc(F)cc(F)c1 44576,C(=O)(C(CCOCCO)NC(=O)CC1CCOC1=O)NCCOCC 44577,c1(C(=O)NC2C3CN(C(CSCCCC)=O)CC32)ncc([N+](=O)[O-])cc1C 44578,N1(C(C(COC)O)=O)CCC(NC(=O)CC2(C)CC2)C2(CCC2)C1 44579,CC1COCC(CC(N2CCC(CN(C)C(c3cc(F)n[nH]3)=O)CC2)=O)O1 44580,c1(C(=O)Nc2cncc(C(N3CCC(CC(=O)OC)C3)=O)c2)cc(Cl)ncc1I 44581,c1(C(=O)NCC2CCCCN(C(C3(C(F)F)CCC3)=O)C2)ccc2nccn2c1 44582,c1(SC)nc(C)c(CCC(=O)N(C2CCN(C(=O)C(C)C#N)C2)C(C)C)c(O)n1 44583,c1(C(N(CCC(C)NC(c2cc(CC)c(CC)o2)=O)C)=O)cc2ncccc2o1 44584,C(=O)(CCS(=O)(=O)NC(C)=O)NC1C(NC(C2N(CCC)CCCC2)=O)CCC1 44585,Cc1cc(Br)cc(C(N2CC(NCc3cccc([N+](=O)[O-])c3)C3(CC3)C2)=O)c1C 44586,C1(C(=O)NCC(COCC)O)CCN(Cc2nnnn2-c2ccco2)CC1 44587,N1(C(C2CC(C)(CC)C2)=O)CC2(CCCC2)C1C(=O)NOCCF 44588,C1(CNC(C(CC)(C)C)=O)CC2(CO1)CN(C(c1cccc(CO)c1C)=O)C2 44589,C(=O)(C(C)(C)C(F)F)N1C(CCNC(CC(C)NC(=O)OC(C)(C)C)=O)CCC1 44590,CCC(C)(CNC(c1nc(C)ncc1Cl)=O)C(=O)Nc1ccc(SC(F)F)cc1 44591,C1(NC(C=C(C)C2CCCCC2)=O)C(CNC(c2csnn2)=O)CCC12CCC2 44592,C1(C(=O)NC(CCC)CCCNC(=O)CSS(C)(=O)=O)CC(C(C)(C)C)=NO1 44593,C1(CC(=O)NCC(CNC(C(C)C2CCC2)=O)O)COC(C)(C)C1 44594,N1(C(C)=O)CCN(C(=O)NC(c2ccc(C)cn2)C)CC1CO 44595,C12(C(N3CC(CNC(C4(C=C)CCCCC4)=O)C(C)C3)=O)C3CC(CC13)C2(F)F 44596,Cc1nccc(Cl)c1C(=O)NC1CN(C(C23CCC(C(F)F)(CC2)C3)=O)CC1O 44597,c1(CC(N2CCCC(NC(C3C(C)CCC3)=O)CC2)=O)ccc(F)c(Cl)c1F 44598,CC1CC(NC(=O)CN2CCCNC2=O)CCN1C(C1CC(=O)N(C)C1)=O 44599,CC1(C)OCC(CC(C(=O)Nc2cccc(C(=O)N(C)C)c2)N2CCCCC2)O1 44600,N1(C(c2ccc(OC)nc2)=O)CCC(NC(=O)C(F)=C2CCC2)C(C)(C)C1 44601,N1(C(c2cnc(CC)o2)=O)CCC=CC1C(=O)NCC(C#N)CC 44602,C(=O)(C1=CCC2CCC1N2C(=O)C(C#N)C(C)(C)C)NCC(C)CCO 44603,N1(C(C)C(=O)Nc2cc([N+](=O)[O-])ccc2F)CC(C)OC2(CCCCC2)C1 44604,C(=O)(CCCN=[N+]=[N-])NCC(C)(O)CNC(C1CCCN1S(C)(=O)=O)=O 44605,Cc1cc(Br)c(F)cc1NC(c1cncc(C(F)(F)CF)c1)=O 44606,c1(OCC(=O)NC(C)CC2CCC(=O)N2)ccc(Cc2ccccc2F)cc1 44607,C1(C(=O)NCCOCCCNC(CC=CC=C)=O)OC(C)CC1C 44608,C#CCCCCC(=O)NCc1nc(C(=O)NC(C)(C)C(O)CO)c(C)o1 44609,C(C#CC(=O)N(CCCCO)CC)NC(C1C(=C)C1)=O 44610,CC12CC(C(N3C4CCC3CN(C(C3C5CCCC35)=O)CC4)=O)(C1)C1(CCC1)O2 44611,C(=O)(C(O)C(C)CC)N(C(CNC(C=CC(=O)OCCCC)=O)C1CC1)C 44612,C(=O)(C1=NN(C)C(=O)CC1)NCCc1cc(C(N(C2(C)CC2)C)=O)no1 44613,C1(C(=O)NC2CCN(C(C3(C#C)CC3)=O)CC2)CN2CCC1(C)CC2 44614,C(=O)(C1=NOC(C)C1C)NC1CN(C(COCCOC)=O)CC1(F)F 44615,c1(C(=O)NC2CCC(C(=O)OCC)C2)ccc(NC(C)(C)C)cc1 44616,C1(NC(C2C(OC(C)=O)C2)=O)CCC(C)N(C(C2CC(C)(C)C2)=O)C1 44617,C(=O)(C#CC(C)(C)C)N1CCC(N(C(c2c(OC)nsc2)=O)C)CC1 44618,c1(N(C(=O)NCC(C(=O)NC)C)C)cc(Cl)c(OC)cc1OCC(F)(F)F 44619,c1(C(CNC(CCN(C)CCO)=O)NC(C2(Cl)CC2(F)F)=O)ccccc1F 44620,O(NC(=O)C(F)(F)C(C)(C)O)C(CC(C)C)C(N1CC2CC=CCC2C1)=O 44621,C(N=c1[nH]c2ccc([N+](=O)[O-])cc2s1)C1(CCNC(C2CCC(C)(C)C2)=O)CC1 44622,c1(C(=O)NCC(CNC(C(C(C)OC)N(C)C)=O)CO)cc(C#N)cn1C 44623,N1(C(c2cccc(SCCC)c2)=O)CCN(C(=O)C(C)COC)C(CC)C1 44624,Cc1cc(Cl)ncc1NC(C1CCCCN1C(=O)Cn1ccc(C)n1)=O 44625,CCCCCC(=O)N1CCCC1(C)CNC(C1(F)CCN(C(C)(C)C)C1)=O 44626,CCC(C)(C)CCCC(=O)NC1(CNC(=O)CC2CCC3CC2C3(C)C)CCC1 44627,c1(C(=O)NCC2C(NC(c3c[nH]cc3Br)=O)CCC2)cc2nn[nH]c2cc1F 44628,Cc1ccc(C(O)C(N2CCC(F)(CNC(c3cc(C#N)c[nH]3)=O)C2)=O)cc1 44629,N#Cc1cc(C(=O)NCCC2CCN(C(=O)COc3ccc(F)cc3)C2)no1 44630,C1(CC(=O)NC)CN(C(c2cc[nH]c2C)=O)CCN1C(=O)C=Cc1cccnc1 44631,C12CCN(CC1(C)C)c1nnc(n1CC1CC1)C2.c1(OC)ccsc1S(C)(=O)=O 44632,c1(OCC)ccc(C(=O)NCC(C)CN(C(=O)C(C)OCCC(C)C)C)cc1C 44633,C1(CC(=O)NCC(C)(C)OCCNC(C2(SC)CCC2)=O)C(C=C(C)C)C1(C)C 44634,C(C)(C(C(=O)NCc1cc(O)ns1)NC(c1nonc1C)=O)OC 44635,c1(C(N2CCN(C(C3C(=C)C3)=O)C(C)C2)=O)cccc2nc(O)[nH]c12 44636,c1(CN(C(=O)NCC(CO)OC)C)nccnc1CO 44637,C(=O)(C(=O)C(F)(F)F)NCC1C(C)(C)C1(C)C 44638,N(C1CCCc2n[nH]cc21)C(C1N(C(CN2CCC(OC)C2)=O)CC(O)C1)=O 44639,c1(C(=O)OC)ccnc(C(=O)NC2CN(C(=O)Cc3ccnc(Br)c3)C2)c1 44640,c1(C(N2CCN(C(C3CC(C)C3)=O)CC2CO)=O)cncc(S(N)(=O)=O)c1 44641,c1(CC)cc(NC(=O)C(CNC(c2cnc(C)s2)=O)OC)cc(O)c1 44642,C1(C(C)=O)CCN(C(=O)CNC(=O)C(C)C)CC1.c12csc(n1)NC2=O 44643,C(=O)(C1Cc2ccccc21)N1CCC(C)(NC(c2n[nH]c(CC)c2C)=O)CC1 44644,c1(SC)ccc(C(=O)NC2CC2CNC(C2CC(C)(O)C2)=O)cc1 44645,C1(NC(C2C(NC(C=CC(=O)N(C)C)=O)C=CCC2)=O)CCCN(C)C1=O 44646,c1(C(=O)NCCC2N(C(CCOCC(C)C)=O)CCC2)ccc(NCCO)cc1 44647,CC1(C)OCC(CCC(=O)NC2CC2c2cnn(-c3ccccc3)c2)O1 44648,C1(C(N(CCCC)CCCC)=O)CCCCN1C(C1CCC2CC12)=O 44649,C1(C)(NC(CC(C)c2cccnc2)=O)CCCN(C(c2cnc(O)n2C)=O)C1 44650,C(=O)(C(C)(C)CC(C)C)NCC1(OC)CCN(C(C2(C)CC2C(F)(F)F)=O)CC1 44651,n1(C(C)C)ncc(Cl)c1C(=O)NC1CCC(C)(CN)C1 44652,c1(OC)c(C(=O)NCC2(F)CC(CNC(=O)C3=CCCC3C)C2)cc(Cl)cc1Cl 44653,Cc1nc(C)c(C(N2CCC(C)(CNC(c3scnc3C3CC3)=O)C2)=O)[nH]1 44654,N1(C(C(C(C)C)SCC)=O)CCN(C(C2CC(C)CCO2)=O)CC1CC(F)F 44655,Cc1cc(C(N2CC=CC(NC(C3(C(N)=O)CC3)=O)C2)=O)c2c(c1)CCC2 44656,C12(C(=O)NC3CC(C(F)C(=O)NCCCN4CCCC4=O)C3)CCC(CC1=O)C2 44657,N1(C(c2cc(-c3ccccc3)no2)C(=O)NC(CC)(C)C)CCC(C(F)F)CC1 44658,C(=O)(C1=CC(O)C(NC(=O)C2=CCCCCC2)C1)NCC1CCN(C(C)=O)C1 44659,C1(C(N2C3CC(CNC(C(COC)C)=O)C2CC3)=O)Cc2ccccc2C(=O)O1 44660,N1(C(C(C2CCCC2)NC(C)=O)=O)CC(C2CN(C(C3(O)CC(C)(C)C3)=O)C2)C1 44661,C1(NC(Cc2cc(OC)no2)=O)CCCCN(c2nnc(-c3ccon3)s2)C1 44662,n1(CC(=O)NC2(C)CC(NC(c3n[nH]cc3Cl)=O)C2)ccc2ccc(F)cc12 44663,S(=O)(=O)(CC(C)C)NC(=O)NCC(C=CC)(O)CO 44664,C12(NC(c3ccc(CC)nc3)=O)CC(CNC(=O)Cc3[nH]cnc3C)(C1)OC2C 44665,CN1CC(O)CC1(C)C(=O)NCC(C)(C)NC(c1cc(C#N)cs1)=O 44666,N1(C(C2(C)CCCCO2)=O)CCN(C(=O)CNC(c2ccncc2)=O)C(CO)C1 44667,c1(C(C(=O)NC(C)C)NC(c2c(C)n(C3CC3)nc2)=O)ccc2c(c1)C=CCC2 44668,N1(C(c2csc(C(F)F)c2)=O)CC2(CCN(C(c3sccc3Cl)=O)C2)C1 44669,C1(C(C(=O)NCCC(=C)C)F)CCN(C(=O)C=CCCC)C1 44670,CC(C)(C)C(CO)C(=O)NC1CN(C(c2cnccn2)=O)C(C)(C)C1 44671,C(C(CNC(c1ccccn1)=O)S(C)(=O)=O)NC(C(C=C)C)=O 44672,C1(NC(C2CCCC(F)C2)=O)CCN(c2nccc(CO)n2)C12CCC2 44673,C#Cc1ccccc1NC(=O)C(CCC=C)NC(=O)CCCC(C)=O 44674,C(CCCCC(=O)N(C)CCC1CCCN1C)NC(C1CC(C(C)C)C1)=O 44675,Cc1cc(C(N2CC(NC(C3(C)CCC(F)(F)C3)=O)C(C)(C)C2)=O)ncc1CO 44676,N1(C(c2c(OC)nsc2)=O)CC(C(=O)NCCC2CCN(C)C2)CC12CCC2 44677,C1(O)(C(=O)NC2(C3CC3)CCNC2)CN2CCCC1C2 44678,C1(CNC(c2cccn2C2CC2)=O)CCN(C(c2cn3c(n2)CCC3)=O)CC1O 44679,N1(C(C2CCCC(C)CC2)=O)CCCC2(C1)CN(C(c1cccc(F)c1Cl)=O)C2 44680,C(=O)(CC(C)(C)CNC(C1CC=CCO1)=O)NCC(C)(C)C(N)=O 44681,C(CC(=O)NCc1ccc(F)nc1C)(C(C)(C)C)NC(C1CCCN(CC)C1)=O 44682,Cc1cc(S(N)(=O)=O)oc1C(N1CCN(C(=O)COC2CCOC2)C(C)C1)=O 44683,CC1CC(C)(C)CCC1NC(=O)C(=O)Nc1cccc(CN2CCOCC2)c1 44684,C(=O)(C(C)(O)C1CCC1)NCC(C)CN(C)C(C1(Br)CC1)=O 44685,N1(C(CC2(OC)CCC2)=O)CCCCC1C(=O)NC1CC(C)(O)C1 44686,C1(NC(C2CC(C)CN(C(=O)C(O)CC(F)(F)F)C2)=O)CCC2(CCCC2)C1 44687,CC1(C(=O)NCC#CC(=O)NCCCC2CCOC2)CCC(=O)C1 44688,N1(C(COc2cc(C)c(F)cc2)=O)CC2CCN(C(c3csnn3)=O)CC2C1 44689,C1(N(C(c2cc(C)n(C3CC3)n2)=O)C)CN(C(=O)C(C)c2cccs2)CC12CC2 44690,c1(-n2cc(CC3CC(C(N4CCN(C(F)F)CC4)=O)C3)nn2)cnnc(O)c1Br 44691,C(=O)(C(C(C)(C)C)n1cc(C(C)N(C)C)nn1)NC1C(OCC)C2C1CCC2 44692,c1(CCC(N2CC(O)(CNC(C=CSC)=O)C2)=O)c(F)cccc1Cl 44693,C1(CN(C(C2COC(=O)O2)=O)CC)CCCCN1C(C1CC(O)CN1C(C)=O)=O 44694,c1(C(N2CCC(NC(C3C(C(=O)OCC)C3)=O)C2)=O)cc(S(N)(=O)=O)sc1Cl 44695,C1(C(=O)NCC(CN(C(C2CCCC(F)C2)=O)CC)(C)C)CC2(CSC2)C1 44696,N1(C(C=CC(C)(C)SC)=O)CCCC12CCN(C(C1CCN(CC(C)C)C1)=O)C2 44697,N1(C(C2CC(OC)C2)=O)CCN(C(c2ccc(SC)s2)=O)C(C)CC1C 44698,C=C(C)CCCC(=O)NC1(CNC(c2cc(F)ncc2OC)=O)CCCCCC1 44699,Cc1cc([N+](=O)[O-])cc(S(=O)(=O)N2CC3(C2)OC2CCC2(C)O3)c1Cl 44700,C(=O)(C1=CCCSC1)NC1(COC)CCN(C(=O)CC2CC23CC3)C1 44701,c1(C(=O)NCc2c(C3CN(C(c4c(C)n[nH]c4)=O)C3)ocn2)coc(C#N)c1 44702,C(=O)(C#CC(C)(C)CNC(c1cnn(C(C)C)n1)=O)NC(C#C)CC1CC1 44703,c1(CC)ccc(C(N2CC3(C2)CN(C(c2sc(OC)nc2Cl)=O)C3)=O)nc1C 44704,C(=O)(C(C)(C=C)CC)NCCC(=O)NC(CC=C)C(=O)OCC 44705,c1(C(N2C(C)CC(C(=O)NCC3(Oc4ccccc4)CC3)C2)=O)ncc(Cl)cc1F 44706,C=C1COc2c(C(=O)NCCC(C)NC(C3(Br)CC3)=O)cnn2C1 44707,C1(C(N(CC(CN(C(CN(C(C)=O)C)=O)C)O)C)=O)CCCCCN1C 44708,CC1COc2ccc(C(N3CCCCC(CNC(c4ccnnc4)=O)C3)=O)cc21 44709,C1(CC(=O)NC2(CC)CCCCC2)CCCN(C(=O)C(O)C2CC2)CC1 44710,C1(CCOC)(NC(C2C=CC=CC=C2)=O)CCN(C(=O)CCc2cncnc2)C1 44711,c1(CN2CCC(C(N(C3(C)CCCC3)C)=O)C2)ccc(Br)c2cccnc12 44712,C1(CC#C)(C(=O)NCC(O)CNC(c2conc2C2CCCC2)=O)CCCCO1 44713,Cc1cc(=NC(C)c2ccc(Cl)c(F)c2)[nH]c(=NCCN(C)C2CC2)[nH]1 44714,c1(CC(=O)NCCC(CNC(C=C(C)C(C)C)=O)O)csc2c(F)cccc12 44715,c1(OC)cccc(C(=O)NCC2(F)CCN(C(=O)CC3C=CCC3)C2)c1F 44716,N1(C(CC(=O)OC(C)(C)C)=O)CCCC12CCCN(C(=O)C(F)(F)C1CC1)CC2 44717,c1(OC(CC)C)cc(CN2CCC(C(=O)N(C)C(C)C)CC2)ccc1OC 44718,C(=O)(C1CCCc2nncn21)NC1(C)CCN(CCCCC2CCCC(F)(F)C2)C1 44719,Cc1c(CC(=O)NC(C)(C)CNC(=O)C=Cc2cnccn2)ccc(Cl)c1Cl 44720,Cc1noc(C(N2CCCC2CNC(=O)C(C2CCCO2)C2CC2)=O)n1 44721,Cn1cc(C(C(=O)NC2CCC2(C)C)NC(=O)Cc2cn[nH]c2)nn1 44722,CS(=O)(=O)c1cccc(C(N2CCCC2CCCNC(C2CCC3CC23)=O)=O)c1 44723,C1(CC(=O)NC(CN(C(=O)CNC(c2ccc(C)s2)=O)CC)C)CC2CC1C2 44724,N1(CC#C)CCC2(CC1)CC2(C)C(=O)NC(c1cccc(Cl)c1)C 44725,c1(OC)cc(C(N2CC(F)CC2CNC(=O)Cc2cc(Cl)cs2)=O)ccc1Cl 44726,Cc1cnc2nc(C(=O)NC3(C)CCN(C(c4cc(C)nnc4O)=O)C3)nn2c1 44727,Cc1cc(C)nc(SCC(=O)NC(C)C(CO)NC(C2(F)CC=CCC2)=O)n1 44728,C=CC1CN(C(C2CC3(CCC3)C2)=O)CC1NC(c1cn(CC)nc1C)=O 44729,C1(C(N(CC(C)C#N)C2CC2)=O)CCN(C(c2ccco2)=O)CC1 44730,n1(CC)cc([N+](=O)[O-])c(C(=O)N(CC(C)NC(=O)Cc2cc(C)cs2)C)n1 44731,C1(NC(C(C)SCC)=O)CN(C(c2cnn(CC3CCC3)c2)=O)CCC1F 44732,C#CCC(C)(C(=O)NC(c1nn(C)cc1O)C)NC(=O)C(C)=C1CCC1 44733,c1(C(=O)OCc2cccc(C(F)(F)F)c2F)nnn2c1COCC2 44734,Cc1ccc(C(F)CC2CCN(C(=O)C(=O)NCCC3CCC3)CC2)cc1C 44735,CN1C(=O)NCC1C(=O)NCCOCCNC(C1OC2CCC1C2)=O 44736,N1(C(C(CC)=CCCC)=O)CCN(C(C23CC(C)C2C3)=O)C(c2nccn2C)C1 44737,C1(C)(CCNC(C2CCC(C)O2)=O)CCN(C(c2cnccc2Cl)=O)CC1 44738,c1(OC)c(Br)ccc(F)c1CN1CC2CC2(C(=O)Nc2cncnc2C)C1 44739,C(CCO)(CC(C)C)NC(c1cc(CNC(c2cc(COC)no2)=O)nn1C)=O 44740,C1(C(N(C)CCNC(=O)Cc2csc(Cl)c2)=O)CCC(CC2CCCCC2)CC1 44741,C(CCS(=O)(=O)C(C)(C)C)NC(=O)NC(c1cccs1)CC 44742,c1(C(N2C(C)C(NC(C3CCC=CO3)=O)CCC2)=O)cc2ccccc2s1 44743,CCC1=C(C(=O)N2CCN(C(c3c(CC)cccc3F)=O)CC(O)C2)CCCO1 44744,C1(C(=O)NCC(C)(C)CCNC(=O)C(O)C(F)(F)F)CCCC2(CCC2)O1 44745,C#CCCCC(C)C(=O)N1CCCC1(CNC(c1cnc(COC)s1)=O)COC 44746,C(C(C)(F)C(C)(C)F)NC(C1CC(C)N1C(c1ncccc1O)=O)=O 44747,C(=O)(CC(Cc1cccc(F)c1)NCc1cnc(-c2ccco2)s1)OC 44748,c1(OC)cc(CCNC(=O)C(C)Cc2ccc(Cl)c(Cl)c2)cc(Br)c1 44749,c1(C(N2C(C)C(NC(c3csc4cncn34)=O)CCC2)=O)cccc2oncc12 44750,S(=O)(=O)(c1ccc(C#N)c(NCC2CCCC(C)(C)CC2)c1)NC(C1CCC1)C 44751,Cc1cc(NC(=O)C(=O)NCC2C3CCC(F)(F)C23)ncc1Br 44752,N1(C(C2CNC(=O)O2)=O)CC2CCCC1C2Cc1cn(-c2c(F)cccc2Cl)nn1 44753,Cc1ccc(F)c(N)c1C(N1CCN(C(=O)CC2CC3(CCC3)CO2)C(C)C1)=O 44754,C(C(=O)N1CC(O)CC1CC(=O)NC1CC(CO)C2CC12)(C(C)C)SCC 44755,N1(CCNC(C2(CC=C)CCC2)=O)CCN(C(=O)C=CC2CCCC2)CC1 44756,N1(C(C2(C(=O)OC)CC2C(F)(F)F)=O)CCN(C(=O)CCC(C)C)CC1C1CC1 44757,N1(C(N2CCCCC2)=O)CC2(CCC2)CC1NC(C(C)(C)NC(=O)C(F)(F)F)=O 44758,C(C(CO)C(F)(F)F)NC(c1sc(Cl)cc1Br)c1n(CCOC)nnn1 44759,N1(C(=O)COCC2CCC2)CCOCC1CNC(C1(CO)CCCO1)=O 44760,N1(C(C2CCC(=O)N2)=O)CC2CCN(C(c3ccc(-c4cccs4)o3)=O)CC2C1 44761,N1(C(C(C=C)c2ccccc2)=O)CCC(CC)C1CNC(c1cnc(S)n1C)=O 44762,Cc1c(C(=O)NC2CC2NC(=O)Cc2cncs2)ccc2c1OC(F)(F)O2 44763,C12(CNC(CCC(=O)N(C)C)=O)CCCCC1N(C(=O)C(=O)C1CCCC1)CC2 44764,c1(C(N2C(CC(=O)NCCCCOC)CCCC2)=O)cccn2ccnc12 44765,N1(C(CSCC(C)C)=O)CC2CCC(C1)N2C(c1c[nH]nc1C(=O)O)=O 44766,C1(NC(CCNC(C)=O)=O)C=CCN(C(=O)Cc2ccc(OCC#N)cc2)C1 44767,N1(C(CC(=O)OCC)=O)CC(NC(c2ccc(C(C)C)o2)=O)CC2(CCC2)C1 44768,C1(NC(c2c(C)nn[nH]2)=O)CN(C(=O)CCN(C)C)CCC1F 44769,Cc1nnc2n1CCC(NC(c1ccsc1Br)c1nnnn1C1(C)CC1)C2 44770,Cc1ccc(-n2nnc(C(=O)NCC3(F)CN(C(C4CSC4)=O)C3)c2C)cc1 44771,C1(CNC(c2n(C=C)ncc2)=O)CC(C)(C)CN1C(c1cc(C#N)oc1C)=O 44772,C1(NCCN(C(C(=O)NCCOc2ccccc2)C2CC2C#N)C)CCCCC1 44773,C#CC1CN(C(c2sc(Br)cc2C)C(=O)NC(C)(C)CC)CC1O 44774,CC1CN(C(=O)CNc2ccccn2)CC(C)N(C(=O)C=Cc2cccnc2)C1 44775,N1(C(C(C=CC)O)=O)CCC=C(C(=O)NC2CCCCCC2)C1 44776,c1(C(=O)NCC2(CNC(C3(C#N)CC3)=O)CCCCC2)ccc2nnn(O)c2c1 44777,N1(C(c2ccc(OC)s2)=O)CC2(CNC(c3snnc3C)=O)CCC1CC2 44778,c1(NC2C(NC(c3c(C)cc(C)o3)=O)CS(=O)(=O)C2)ncc(S(C)(=O)=O)cc1Cl 44779,C(C(=O)NCCC1CCN(C(=O)C(CC)N(C)C)C1)(C(C)C)NC(COC)=O 44780,C=CCC(F)(F)C(=O)N1CCCC1CCC(=O)NCc1ncoc1C 44781,Cc1cc(C(C)NC(N2CCCC2C2CCCOC2)=O)cc(C)c1 44782,N1(Cc2c(C)nncc2)CC2CC1CN2C(=O)CC(=O)N(C)C 44783,C1(NC(c2ccc(SC)o2)=O)CCN(C(c2cnc(NC3CC3)s2)=O)CC1CO 44784,c1(C(N2CCN(C(C(CCC)=CCC)=O)CC2C2CC2)=O)ccc(C#N)cc1C 44785,O=C(C1=CC2CC=CCC12)NCC=CCNC(C1(O)CC(F)(F)C1)=O 44786,C1(F)(CNC(=O)C=C(Cl)Cl)CCC(NC(c2cccc(C(F)(F)F)n2)=O)C1 44787,C1(NC(CC2C(NC(=O)CSc3ccc(O)cc3)CC2O)=O)CCC(F)(F)CC1 44788,c1(C(N2C(C(=O)Nc3c(C#N)cc(Cl)cc3)CCCC2)=O)cc2cc[nH]c2cn1 44789,CC1CCC(NC(c2ccc(Cl)c(C(F)(F)F)c2)=O)CN1C(c1cnnn1C)=O 44790,N1(C(C(F)=C(C)C)=O)CCCCC2(CCN(C(c3ccn(CCO)c3C)=O)C2)C1 44791,C1(C(=O)NCCCCCNC(C(C)OCCOCC)=O)CC2CC1CC2(F)F 44792,N1(c2nc(N3C4CS(=O)C(C4)C3)nc3c2CCC3)C2CCC1c1cncnc1C2 44793,c1(C(=O)NCC(C)NC(C(C2CCCCC2)OC)=O)c(C)cc(Br)cc1C 44794,N1(C(C2(C)CCNC2=O)=O)C2CCC(C2)C1C(=O)Nc1cnccc1N(C)C 44795,CC1(C)CCOC1CCNC(=O)C(N1CCC12CNC2)=O 44796,C1(NC(COc2cc(C)on2)=O)CN(C(=O)C(C)C2CC2)CC1C(F)(F)F 44797,CC1(C(=O)NC(CCCNC(=O)C=CCO)c2ccccc2)CCC(=O)N1 44798,CC(N=[N+]=[N-])C(=O)N1CCCC1C(C)NC(C1C2CCCOC12)=O 44799,CC(C)(Cc1cnn[nH]1)C(=O)NCCCOC1CCOCC1 44800,C1(NC(C(C)Cn2ccnc2)=O)CC2(CCN(C(=O)C3=CCCC3)CC2)C1 44801,C1(OC)CCC(NC(=O)C(CC2CC2)NC(c2csc(Cl)c2)=O)C1 44802,C1(OC(C)=O)CCN(C(=O)NCC2(C)CSC(C)=N2)C1C 44803,C1(O)(CCNC(c2cc(C(F)(F)F)cc(O)c2)=O)CCCN(C(=O)C=CBr)C1 44804,c1(OC)c(C(=O)NCC2CCN2C(=O)C(F)n2ccnc2)csc1C 44805,C(=O)(CC1=NN(C)C(=O)C1)N1CCC2(C(NC(C(CSC)OC)=O)C2)C1 44806,c1(NCC2CCC(NC(c3cn(CC)nn3)=O)C2)ncc2cccnc2n1 44807,N1(CC2(C)CCC2)CCC(NC(=NCC2CCCO2)NC2CCCCC2)CC1 44808,N#CC1(C(=O)NC2CCCC2NC(=O)C2=CCCSC2)CC12CCCC2 44809,c1(OCC(=O)OC)ccc(S(=O)(=O)NC(C)(C)CCC(=O)O)cc1OC 44810,n1(CC)cc(Br)c(CC(=O)NCCNC(=O)Cc2cncs2)n1 44811,CC(CCN(C)C)C(=O)NCc1ocnc1C(=O)NCC(C)C#N 44812,c1(CC(C)NC(C)C(c2ccccc2F)O)ccc(C(F)(F)F)cc1[N+](=O)[O-] 44813,C1(C(C)C)CCCN(Cc2cn(-c3ccc(Cl)cn3)nn2)C1 44814,Cc1ccc(S(C)(=O)=O)cc1C(=O)NCCCCC(C)NC(C1(F)CC1)=O 44815,c1(NC(C2CC(NCc3cc(C(=O)O)cc(Br)c3)C2)=O)nccc(Cl)c1Cl 44816,O=C(CCS(=O)(=O)Cc1ccccc1)NCCC1CSCCN1C(C1CCC1)=O 44817,N1(CCC)CCCC1C(=O)NCC(C)NC(c1cnc(-c2ccsc2)s1)=O 44818,c1(C(=O)NCC2CC(NC(CC3CCC(C)C3)=O)C2)csc(=NC2CC2)[nH]1 44819,c1(OC)cc(OC)cc(C(=O)NC(CNC(=O)CC2CC23CC3)CCOC)c1 44820,C1(C(NOC(CC)C)=O)CN(C(C2CC3CCCC3C2)=O)CCN1C 44821,N1(C(Cc2ccc(OCC=C)cc2)=O)CCC(NC(c2cc(C)ns2)=O)C(F)C1 44822,S(=O)(=O)(c1ccc2[nH]c(=NCC(C)(C)C(F)F)sc2c1)NCc1c(OC)nsc1 44823,c1(C(N(CC(C)N(C)C(c2c[nH]nc2Br)=O)C)=O)ccc(O)cc1F 44824,n1(CC)c(C(=O)NC(C)C(C)NC(c2ccoc2Cl)=O)nc2ccccc12 44825,N1(CC(CC)Oc2cccc(F)c2)CC2CN(C(C3C4COCC34)=O)CC2C1 44826,c1(CC(=O)N(c2cc(C3CCC3)[nH]n2)Cc2ccccc2)ccccc1F 44827,C1(CC(=O)N(C)Cc2nnc(CC)o2)CCCC(NC(c2cscc2C)=O)C1 44828,c1(C(N(C2CCCC2)CCCNC(C2CC(=C)C2)=O)=O)cc([N+](=O)[O-])sn1 44829,C#CCC(C)(C(=O)NCC(=O)NCCOOC)NC(=O)C(C)OC.C1CCCC1 44830,c1(C(=O)OC)cccc(CC(C)C)c1.CCC1CNC(=O)N1 44831,N1(C(C(C(COC)C)C)=O)CCCC2(C1)CN(C(=O)COc1cccc(F)n1)C2 44832,c1(CC(N2CCC(CN(C(c3cn(CC)nc3C)=O)C)C2)=O)ccc(C)cc1C 44833,c1(C(N2CCCC(CCNC(CC(C)SC)=O)C2)=O)cnn2c1S(=O)(=O)NCC2 44834,c1(C(N2CCC(C(C)NC(c3cc(C)n(C(C)C)n3)=O)C2)=O)cccc(N)c1C 44835,N1(C(CC2CCC(C)(C)O2)=O)CCC(C(=O)NC2CC2)CC1(C)C 44836,C1(C(N2C(C(=O)NCCCC(C)O)CCCC2)=O)CC2CC1CC2O 44837,N(C)(S(=O)(=O)N1CC2CC(O)CC(C2)C1)CCCC 44838,N1(C(c2ncnc(C)c2C)=O)CCCC2(NC(C34CC(F)(C3)C4)=O)CC2C1 44839,N1(C(C)=O)CCc2cc(C(=O)N(CCCNC(C3CCNC3=O)=O)CCO)ccc21 44840,C1(CNC(CNS(NC)(=O)=O)=O)CN(C(c2ccc(C)nn2)=O)C2CCCCC12 44841,C(=O)(CCCC(CC)NC(=O)CCC1CCCC1)NC(C#C)(C)C1CCC1 44842,C(=O)(C#CC(C)(C)CNC(=O)C(=O)NCC(F)F)N1CC(C)OCC1 44843,N1(C(C(C)N(C)C)=O)CCCC1(C)CNC(C1CCCC2CC12)=O 44844,c1(SC2CCC(C(N(CCCC)CC)=O)CC2)cccc(S(N)(=O)=O)c1 44845,c1(-c2nnn(CC(N3CCCC3C3CC3)=O)n2)ccc(Br)cc1 44846,N1(C(Cc2nn(C)c(Cl)c2)=O)CCC(C2CN(C(=O)CC(=O)NC3CC3)C2)CC1 44847,C1(CNC(c2ccc(C)o2)=O)N(C(c2ccc(F)c(Cl)c2)=O)CCC1(C)C 44848,Cc1nc2nccc(C(N3CC(NC(C4(N(C)C)CCC4)=O)C(F)C3)=O)n2n1 44849,N1(c2nnc(C)o2)CCCCC(NC(c2nnn(C(C)C)c2C)=O)C1 44850,N1(C(Cc2ccn(C)n2)=O)CCC(CO)(CNC(C2CCCC23CC3)=O)CC1 44851,S(=O)(=O)(c1ccc(NCCCS(C)=O)c(C#N)c1)N(CC)CC1CC1 44852,c1(C(=O)NCCN(C(C(C)=C2CC2)=O)C)cccc(SC(C)C)c1 44853,Cc1ccc(C(=O)NCc2nc(C(=O)N(C(C)(C)CO)C3CC3)c(C)o2)cn1 44854,c1(C(=O)NCC(C(C)C)NC(=O)C(F)C2CCCC2)cnn2cccnc12 44855,CCC(CC)C(C(=O)NCC(C(C)(C)C)NC(c1cc(O)nn1C)=O)OC 44856,CCC(C(=O)NC(C1(O)CN(C(c2cc(C)cs2)=O)C1)C)N(C)C 44857,N1(C(C2C(=C)C2)=O)CCC2(NC(=O)COc3ccccc3OCC)CC2C1 44858,CCC(CNC(=O)CNC(c1ccccn1)=O)(CC)NC(=O)C(C)C#N 44859,C(CCC(O)C(=O)N1CCCC(O)C1)NC(c1c(CC)ocn1)=O 44860,O=C(O)CC(C(=O)O)NC(C12CC(n3cc(-c4ncccn4)nn3)C1C2)=O 44861,c1(C(=O)NC2(C)CCCN(C(C(F)=CC)=O)C2)ccc(C(F)(F)F)c([N+](=O)[O-])c1 44862,Cn1nnc(C(=O)NCCCC(C)(C)NC(C2CC3(CC3)C2)=O)c1C(F)F 44863,C(=O)(C1=CCCSC1)NCCn1cc(C(=O)NC(CCCC)CC)nn1 44864,O=C1C2CC3C1C3(C(=O)NCCc1nc(C(=O)O)no1)C2 44865,Cc1cn2c(n1)CC(C(=O)NC(C)CC1CN(C(=O)CNC=O)C1)CC2 44866,n1(CC(=O)N(C2CCN(C(CC(C)(F)F)=O)CC2)CCO)ccc(O)nc1=O 44867,c1(-n2cc(COCC3CN(C(C4CC4(Br)Br)=O)C3)nn2)cnccc1C(F)(F)F 44868,C(=O)(CCCS(N)(=O)=O)NC(C1OCCN(C(c2ccc(CC)cc2O)=O)C1)C 44869,c1(C(=O)NCC(C(C)(C)C)NC(c2c(OC)cncc2)=O)n[nH]c2c1CCOC2 44870,Cn1nc(Br)cc1C(=O)NCC1CCC(NC(C2OCCO2)=O)CC1 44871,C1(C(C(=O)N(CCNC(c2ccc(C(C)O)cc2)=O)CCO)O)CCC(C)(C)CC1 44872,CC1CN(C(c2cncn(C)c2=O)=O)CCC1N(C)C(c1ccc([N+](=O)[O-])[nH]1)=O 44873,C(C)(CCC(=O)NCCCC1(NC(=O)COCc2ncccc2Cl)CC1)OC 44874,C1(F)(CNC(c2n(C)ncc2)=O)CCCN(C(C2CC(=O)N(CC3CC3)C2)=O)C1 44875,N1(C(C(C)OCCCC)=O)CCCC(CCNC(C2(O)COC2)=O)C1 44876,C1(N(C(COCC(=O)NC)=O)C)CCC2CN(C(C34CCC(CC3F)C4)=O)CC12 44877,N1(C(c2ccc(O)nn2)=O)CCN(C(c2ccnc(-n3cccc3)c2)=O)C2CC12 44878,N1(C(c2c(CNC(C(CCSC)O)=O)cnn2C)=O)CCN(C)C(=O)C1 44879,C(=O)(CCCC(F)(F)F)NC1CC(N(C(=O)C(C2CCCCCC2)F)C)C1 44880,c1(CCC(=O)OCC)nc(O)c2c(C)c(C)sc2n1.C1(=O)C(C)N1C(CC)=O 44881,C1(CNC(C2(CC)CN(C(C3CCC(CO)CC3)=O)C2)=O)CC2C(C1)C2(F)F 44882,C12(CNC(CC(C(C)C)C)=O)CCC(NC(=O)COC(F)F)(CC1)CO2 44883,N1(C(C2(NC(CCCOC(C)=O)=O)CCSC2)=O)CC(CO)C(C2CC2)C1 44884,C1(CC)(NC(=O)C(C)(F)F)CCCN(C(C2CC(C)(C)CN2C)=O)C1 44885,C1(CN(C(C(C)C2CCOC2)=O)C)CCCN1C(=O)CCc1cnn[nH]1 44886,C12(C(C)NC(C(COCC)NC(C3CC(F)(F)C3)=O)=O)CCC(CC1)C2 44887,C(=O)(CC(C(F)F)NC(c1ccco1)=O)NC(CN(C)C)CO 44888,N1(C(=O)Nc2nc(=N)s[nH]2)CCNCC1c1cccc(Cl)c1 44889,c1(C(C)C)ccc(CC(C)NC(=O)CCNc2ccc(-c3ccsc3)cc2)cc1 44890,N1(C(C(COC)(F)F)=O)CCCCC(N(C(=O)Cc2cnn(C)c2C)C)C1 44891,N1(C(CCOC)=O)Cc2nccn2CC(NC(C23CCC2C3)=O)C1 44892,c1(C(C(=O)NCC2CC(NC(C3C(CC)OCC3)=O)C2)O)ccc(Cl)cc1 44893,C1(C(=O)Nc2cccc(CNC(C(C(=O)OC)OC)=O)c2)CCC2(CC1)CC2 44894,N1(C(C(C2CCC2)NC(C2N(CCC)CCC2)=O)=O)CCC(COC(C)=O)C1(C)C 44895,N1(C(Cc2c(C)nc(C)s2)=O)CCCC(N(C)C(c2cnc(C3CC3)[nH]2)=O)CC1 44896,C(CCC(=O)NOCCCCC)(C(C)C)NC(CCC=CC)=O 44897,N1(C(c2ccc(CC)cc2)=O)CC(NC(=O)COCCSC)C2(CC2)C1 44898,C12(C(=O)NC(C)C(C)NC(c3ccc(O)nn3)=O)CCCN(CCC1)C2 44899,C(CC(C(=O)N(CCO)CCN(C)C)NC(=O)CC(O)c1ccccc1)OC 44900,CCC(C)(CNC(=O)CCC1CCCCO1)C(=O)N(C)CC1(N(C)C)CCC1 44901,O=C(C1=CCOC1)NCC1CN(C(=O)COc2ccc(F)cc2)C2CC12 44902,C(=O)(CCCC(=O)C1CC1)NC(C(=O)NCCc1cc(C)[nH]n1)C 44903,c1(SC)cccnc1C(N1CCC(NC(c2cnc(O)o2)=O)CC1)=O 44904,N1(C(C(CC=CCC)C)=O)CCC2(CCC2NC(c2ccoc2C)=O)CC1 44905,N1(C(C2C(CNC(c3c(CC)n[nH]c3)=O)CCC2)=O)CCCCCCC1C 44906,C(CNC(=O)C(=O)C(C)C)(CC(=O)N(C(CO)C1CC1)C)OC 44907,CCC(C)C(C(=O)NC(CNC(C1CC(C#N)C1)=O)C1CC1)NC(=O)OC 44908,c1(C(=O)NCC23CC2CN(C(=O)Cc2nc[nH]n2)C3)cc2ccc(F)cc2[nH]1 44909,CC(CC(F)(F)F)C(=O)N(CCCCN(C(=O)C(CO)C(F)(F)F)C)C 44910,c1(-c2ccc(C(=O)NC(CCCNC(CS(CC)=O)=O)C)o2)c(C)cccc1C 44911,C1(NC(c2c(C(C)C)onc2)=O)CCN(C(=O)CS(=O)(=O)N(C)C)CC1C 44912,c1(CC(=O)NCC2N(C(C(CC)F)=O)CC=C2)cc(C)cc(Br)c1 44913,CCC(O)C(C)(C)C(=O)NC1CC(C(=O)NCC2(CO)CCN(C)C2)CC1O 44914,C(C1CN(C(c2cncc(F)c2Cl)=O)Cc2ccccc21)NC(C(N)=O)=O 44915,c1(CC2CC(c3ccc(-n4cc(C5C(OC)C5)nn4)cc3)C2)cc(F)ccc1F 44916,N1(C(C(C)C2CC2)=O)CCCC1CCNC(=O)CN1CC2CC2C1 44917,CC1CC(NC(=O)CCc2ccccc2O)CN1C(=O)C(N)=O 44918,N1(C(C2N(C(c3cc(COC)[nH]n3)=O)CC(C)C2)=O)CCC(O)C(C)C1 44919,CC1(CNC(=O)C(C2CCC2)NC(=O)Cc2ccccn2)CCCOC1 44920,C1(NC(=O)CCc2cncs2)CC1C1CCCN(C(c2cc(Cl)cs2)=O)C1 44921,C1(C(=O)N(CCC(F)(F)F)CCO)C(CO)C1(F)F 44922,C1(CN(C(C(c2ccccc2)SC)=O)C)CCCN1C(C1CN(C(N)=O)C1)=O 44923,N1(C(C2C(C)CN(C(c3ccc(CO)s3)=O)C2)=O)CC(C)(C)CC1CO 44924,N1(C(C2(C(C)C)N(C(c3cc(C(C)C)no3)=O)CCC2)=O)CCCNC(=O)CC1 44925,O=C(N=c1[nH][nH]c2c1CCCC2)C1CN(Cc2cn3c(Br)cccc3n2)CCS1 44926,N1(C(=O)CC2CCC3CC23)CC23CCCC2(C1)CN(C(c1ccnnc1)=O)C3 44927,N1(C(C(CCCOC)NC(=O)CCC(CF)CF)=O)CCCC2CNC(=O)C12 44928,C(CS(=O)(=O)CC(=O)NC(C)(C)CC(F)C(=O)NCC(CSC)OC)OC 44929,CC(CC(C)(F)F)C(=O)NCC=CCNC(=O)CCCc1nncn1C 44930,c1(C(=O)OC)ccc(NS(=O)(=O)NCC2CC(F)C2)cc1 44931,C(=O)(C(C)Cc1ccco1)NC.c12nc(co1)C(=O)NOC(C1CC1)C(=O)NC2 44932,C=CC(C)(C)CCNC(c1ccnn1C)c1nnnn1-c1ccccc1C 44933,C1(NC(C(C=CCCC)O)=O)COC2(CNC(c3ccc[nH]3)=O)CC1C2 44934,C1(C(=O)NCc2cc(C3CCC3)no2)CCCN(C(=O)C(F)CC2CCOC2)C1 44935,Cc1ccc(C)c(C(=O)NC(C)CC(C)NC(=O)C=Cc2ccc(=N)[nH]c2)c1 44936,N1(C(c2c(C)cccn2)=O)CCCC(C2CC2NC(=O)CCC(F)F)C1 44937,N1(C(C(C)OCCOC)=O)CC(O)(CNC(c2cnns2)=O)C1 44938,c1(C(=O)OC)cc(F)cc(F)c1NCc1cnc(C(C)(C)C)s1 44939,C1(CC=C)(NC(c2ccc(OC)nn2)=O)CCCN(C(c2nsnc2O)=O)C1 44940,C=C1CC(N=c2[nH]c(=NCC(=O)NC3CC3)[nH]c3cc(OC)ccc23)C1 44941,C#Cc1cc(C(N2CC(NC(c3cc(Cl)cnn3)=O)CC(O)C2)=O)cc(F)c1 44942,N1(C(c2cncc(C)n2)=O)CCC(NC(c2ccc(Cl)[nH]2)=O)C1(C)C 44943,C12(NC(=O)Cc3nc(F)c(F)cc3F)CCCN(C(c3cnsc3)=O)CC1C2 44944,C1(C(=O)OC)CN(C(=O)NCc2cnc(O)cc2OC)CCC1C 44945,N1(C(c2cc(C(N)=O)[nH]c2)=O)CC2(CNC(C34CCCCC3C4)=O)CCC1CC2 44946,C(N(CC(C)C#N)N1CCCC(F)(F)C1)c1ccc(C)cc1F 44947,CCS(=O)(=O)c1ccc(S(=O)(=O)N2CCN(C(C3CC3C)=O)CC2)cc1 44948,C1(CC)CN(C(c2cc(C)ncn2)=O)CC1C(=O)NC(CC1CC1)C1CC1 44949,N1(C(COCCCC)=O)CC(CC(=O)N(CCC(N)=O)C2CC2)C2(CC2)C1 44950,c1(CC)ccc(NC(=O)C(C2CCCO2)NC(=O)CC2(C)CCCCC2)c(C)n1 44951,N1(C(CCCCOC)=O)CC2CCCC(CNC(=O)Cc3nnc(C)o3)C2C1 44952,c1(CC)cc(C(=O)NCC(O)CCNC(=O)COc2cccc(F)c2)ccc1C 44953,C(c1ccccc1F)=CCC(N1CC(CCO)(NC(c2cc(C#N)sc2)=O)C1)=O 44954,C(=O)(C1OCCc2c(Br)cccc21)NCCCCN(C(C(CC)C)=O)C 44955,C(=O)(C#CC1CCCCC1)NCCCN(C(C1CCC(C)S1)=O)CC 44956,c1(SC)cc(C)nc(N2CCC(C(C)NC(c3ccc(C(F)(F)F)[nH]3)=O)CC2)n1 44957,CCCCCCC(=O)NC(C(c1ccccc1)NC(c1cc(C)[nH]n1)=O)C(C)C 44958,CC(=Cn1ccnn1)C(=O)N1CC2(CCN(C(c3cc4n(n3)CCO4)=O)C2)C1 44959,CCCCC(CC)CC(=O)NCC(CNC(=O)C(=Cc1cccc(F)c1)F)CO 44960,C1(CNC(CCC)(CC)c2nnnn2C2CCCC2)CCN(C)C(=O)C1 44961,O(P(C)(=O)CCNC(C1SCCCS1)=O)CC 44962,c1(CC)cc(OCC(N2CCCC2CNC(=O)CCCC#N)=O)ccc1Cl 44963,c1(OC)cc(C)ccc1OCC(=O)NC(CNC(c1cn(C)cn1)=O)C(C)(C)C 44964,c1(C(N(C)CC2CCCCN2C(C2CC23CCC3)=O)=O)c(F)cc(F)c(F)c1F 44965,O=S(=O)(c1c[nH]ccc1=NCC1COCO1)NCC1COc2ccccc2O1 44966,Cn1nc([N+](=O)[O-])cc1C(=O)NC(C)(C)CNC(=O)C(c1cncn1C)O 44967,C1(CNC(c2c(C)cns2)=O)CC2(CCN(C(C3COCCN3C)=O)CC2)CO1 44968,C1(C(N2CCCC(N(C(c3c(CC)scc3)=O)C)C2)=O)CCc2ncncc2C1 44969,c1(C(N(CC(C)N(C(C(C)n2cnnn2)=O)C)C)=O)c(O)nnc2c1COCC2 44970,C12(NC(c3c(C)nc(C4CC4)s3)=O)CCN(C(=O)C(C)(C)n3cccn3)CC1C2 44971,C1(NC(c2c(C3(C)COC3)noc2)=O)CCCN(C(=O)Nc2cncc(N)n2)C1 44972,C=CC(F)(F)C(=O)N1CCC1CNC(c1ccc(C(C)(C)C#N)cc1)=O 44973,N#CC1CC12CCN(C(C1(F)CCN(C(C3CCNC3=O)=O)C1)=O)CC2 44974,C12(CNC(CCC(=O)NC)=O)CCC(CNC(C3CC3(C)C(C)C)=O)(CC1)OC2 44975,c1(CC(=O)N(C)C)ccc(C(=O)NCCC(O)CNC(c2cccnn2)=O)cc1 44976,c1(C(C)=O)cncc(C(=O)NC(CNC(=O)CCc2c(C)noc2Cl)CO)c1 44977,N1(C(C2N(C(C)=O)CCC2)=O)C2CCC1C(NC(c1cc(Cl)cnc1C)=O)C2 44978,CC(C)(C)CCCC(=O)N1CCN(C(c2ccc(C#N)cn2)=O)CC(CO)C1 44979,c1(C(C)NC(c2c(Br)cnn2C)c2n(CCOC)nnn2)ccc(F)cc1 44980,c1(OC)nccc(C(=O)NCC2CCCC2NC(C2C3CCCC23)=O)c1F 44981,CC(C)C(O)C(F)(F)C(=O)NC(C1CN(C(=O)C(C)O)C1)C 44982,C1(NC(c2cn3ccsc3n2)=O)CN(C(=O)C(Cl)=CCl)C2(CCCC2)C1 44983,C(CC(C)CC)(C(=O)NC(C)(CC)CCC)NC(CC=CCCCCC)=O 44984,Cc1cc(=NC(C)c2ccc(C)o2)[nH]c(=NCCC(=O)N(C)C)[nH]1 44985,C(C1=CCC2CC1C2(C)C)(c1nnnn1C)Nc1cccc(C(C)F)c1 44986,N1(C(Cc2c(C)noc2)=O)CCN(C(C23CC(CO)(C2)OC3C)=O)C(C2CC2)C1 44987,C1(CCC)(NC(C2CCS(=O)(=O)N2)=O)CCCN(C(c2cnsc2)=O)C1 44988,c1(C(=O)NC(CC=C)CNC(c2c(C)ncnc2O)=O)cnc2n1CCCC2C 44989,N1(C(C)Cc2ccncc2)CC(N(C)C(=S)NCC(F)(F)F)C(F)(F)C1 44990,c1(CNC(C(CC)N(C)C)=O)ccccc1CNC(=O)CC1CC2CC2C1 44991,c1(C(N2CCC(O)C(F)C2)=O)c(C)[nH]c(NCc2c(OC)nccc2)c1C 44992,c1(COC)ccccc1C(=O)N(C(CNC(=O)CCC(=O)OC)C1CC1)C 44993,c1(NCC2C(NC(c3ocnc3C(F)F)=O)CCCC2)ncc2cccnc2n1 44994,C1(NC(CC2(CNC(Cn3ncc(CC)c3)=O)CC2)=O)CCCC1N=[N+]=[N-] 44995,n1(CCC)ncc(C(N2CC3C(NC(C4(C5CCCCO5)CCC4)=O)C3C2)=O)c1C 44996,c1(OCC)cccc(OC(=O)C(C2CCCCC2)NC(C2C3CCCC23)=O)c1 44997,N1(C(c2c(OC)cccc2C)=O)CC2CC3CC2C1C3NC(=O)C=C(Cl)Cl 44998,c1(OC(C(C)C)C(=O)NCCC2CCCN2C(=O)C2CC2)ccc(F)cc1F 44999,N1(C(CONC(=O)OC(C)(C)C)=O)CC2(CCN(C(C34CCN(CC3)C4)=O)C2)C1 45000,c1(CC(=O)NC2C(NC(C3(COCC)CC3)=O)CCC2)ccc(Br)nc1 45001,c1(C(=O)NCCC(C)NC(CCCN(C(C)C)C)=O)c(F)cc(O)cc1F 45002,CC(C)(C(=O)N1CC2CCC(NC(c3ncsc3Br)=O)(C2)C1)S(C)(=O)=O 45003,c1(C(N2CCC(CNC(c3occc3C3CC3)=O)C2)=O)ccc2c(c1)OCCC2 45004,C1(CCC)CCC(C(=O)NCC2(C(N)=O)CN(C(C3NC(=O)CC3C)=O)C2)CC1 45005,CCC(F)(CNC(=O)CC1CCCCN1C(=O)CCCOC(C)=O)CC 45006,N1(C(C2C(c3ccc(C)s3)C2)=O)CCC(C)C1CNC(C1(C)CCC1)=O 45007,Cn1cnc(C=CC(=O)NC2(C(N3CC(c4ccccc4)C3)=O)CSC2)c1 45008,C1(CNC(CNC(C)=O)=O)CCN(C(=O)C(C)Cc2ccc(Cl)cc2)CC1O 45009,n1(CC)nccc1C=CC(N1CC(CNC(=O)Cn2ccccc2=O)C(C)C1)=O 45010,C(=O)(C1=COCCO1)NC1C(C2CCN(C(C(CC)=CC)=O)CC2)OCC1 45011,C1(C(C)NC(c2cc(C3CCC3)[nH]n2)=O)CN(C(C2C3CCC2CC3)=O)CCO1 45012,c1(CC)c(C(N2CC(C)(NC(=O)C(CC)NC(N)=O)C2)=O)csc1C 45013,Cc1nc(C(C)C)ccc1C(=O)NC1(C)CCN(C(C2(F)CCC(C)CC2)=O)C1 45014,Cc1[nH]nc2ncc(C(=O)NC3CN(C(C4CCC(=O)C4)=O)CC3O)cc12 45015,C1(C)(C(N(C(C)CNC(=O)CNc2ncccn2)C)=O)CCC(F)(F)C1 45016,c1(CN(C(C)CNC(c2ccc(N(C)C)nc2)=O)C)c(F)c(F)c(F)c(F)c1F 45017,c1(C(CNC(C2CC=CCO2)=O)NC(C(C)(C)N(C)C)=O)ccccc1F 45018,c1(C(N(C)CC2(O)CCN(C(=O)CSCC(N)=O)C2)=O)oc2ccccc2c1Cl 45019,C1(CNC(CC2CC(C)C2)=O)Cc2ccccc2CN1C(=O)C1=COCCC1 45020,c1(C(=O)NC(C(C)C)CNC(=O)C(C)CF)cccc(N)c1N 45021,N1(C(c2cc(COC)no2)=O)CC(NC(=O)C(O)C2CCC2)CC12CCOCC2 45022,C(CC(C)(C)CC(=O)NCc1nnn(C)c1C(=O)NC1CCN2CCC1C2)OC 45023,N1(C(CSCCNC(C2CC(=O)NC2)=O)=O)CCN2C(=O)NCC2C1 45024,c1(C(=O)NCCNC(C(C(C)C)CN(C)C)=O)cccc2ncnn12 45025,C12(C(=O)NCCNC(C(c3cncnc3)C)=O)C3CCC(CC13)C2(F)F 45026,c1(NC2CCN(CC(=O)NC3CC3)C2)ccc(OC)c(F)c1.N12CCCCC1C2 45027,n1(CC)ncc2c1CCCC2NCCN(CC(O)COc1cccc(C#N)c1)C 45028,C12CC(C1(C)C)C(=O)N2.n1(CC)cnc(C(N2CC(c3csc(C)n3)C2)=O)c1 45029,N1(C(C(CC(C)C)OC)=O)CCC(C)(C)C(CNC(=O)C=CC2CC2)C1 45030,c1(C(=O)NCc2ccc3[nH]ccc3c2)cc2ccc(-c3cn[nH]c3)nc2[nH]1 45031,CC1OC2(CO)CC1(C(=O)NC(C)CN(C)C(C1CC3CCC(C1)C3)=O)C2 45032,C(CCC(c1nnnn1C1CCC1)NCCC1(OC)CCCC1)OCC 45033,c1(CC(=O)NC2(C)CCN(C(Cc3ccn(CC)n3)=O)C2)noc2ccccc12 45034,C1(C2CCN(CCN3CCC(O)CC3)C2)(NC(c2cc(C3CCC3)[nH]n2)=O)CC1 45035,C(=O)(C(CO)NC(C1CC(=C2CCC2)C1)=O)N(CC(C)OC)C 45036,C(CC(F)(F)F)N(C(c1cn(CCNC(c2n[nH]cc2C)=O)cn1)=O)CC 45037,N1(C(c2ccc(C(=O)OC)[nH]2)=O)CCN(C(c2cc(C)ns2)=O)CC(C)(C)C1 45038,CC(Cc1cnc[nH]1)C(=O)OCC(=O)N(C)CC1CCCCC1 45039,C1(NC(c2occ3c2CCCC3)=O)COC2(CCN(C(=O)C3=CCSC3)CC2)C1 45040,c1(C(=O)NC(C2CCOC2)C)coc2c1CN(C(c1[nH]ccc1C1CC1)=O)C2 45041,C(c1ccccc1)=CCOCCN(C(C(C1CC1)OC)=O)C.C1CC1 45042,C1(CC)CC(O)CN1C(c1csc(C)c1)C(=O)NC1CCCCC1 45043,N=c1[nH]c2ncc(C(=O)NCC3CCCN3C(=O)COC3CC(F)(F)C3)cc2s1 45044,Cc1occc1C(=O)NCCc1cc(C(=O)NCC(C)(C)C#N)no1 45045,C(=O)(C(CCSC)NC(c1cccnn1)=O)NCC(=O)NCC=C 45046,O=C1CCC(CCC(N2CCCC2CNC(=O)CC2CSC2)=O)N1 45047,C1(SCCN2CCN(C)CC2)CCOCCN1C(c1cc(F)ccc1N)=O 45048,C1(C(N2CCC(CC#C)C2)=O)(NC(=O)CC(C)(O)COC)CCC(C)(C)C1 45049,N1(C(Cn2ncc(CC)c2)=O)CC(C)CC1C(=O)N(C(C)CSC)C 45050,c1(CN(C(=O)CN2C(C)CCCC2C)CCOC)ccc2ncc(=O)[nH]c2c1 45051,c1(C(=O)NC(CNCC)C)ccc(OCCF)cc1.C1(CC(=O)N)CC2CC2C1 45052,N1(C(c2cc(C)[nH]c2)=O)CC2CCC1C(CNC(c1cccc(F)c1Br)=O)C2 45053,CCCCC(C(=O)NCCCC(C)(C)NC(c1cccc(CF)c1)=O)NC(N)=O 45054,C(CC(O)CNC(=O)CNC(=O)C(F)(F)F)NC(CCSCCC)=O 45055,c1(NC(c2c(C)cc(I)cc2)=O)ccc2c(c1)ncn2C 45056,C1(C)(COCCC(=O)NCC=CC)COCC(C)(C)O1.C12CC1SCCNC2=O 45057,N1(C(Cc2c(C)nc[nH]2)=O)CCC(NC(c2sc(F)cc2Cl)=O)C(CO)C1 45058,C(CC(C)(C)C#N)(C(=O)NC1CCCCC1)N(C(C)C(C)n1cncn1)C1CC1 45059,Cc1nc(C(N2CCC(OCCNC(c3ccnnc3)=O)C2)=O)n[nH]1 45060,C1(C(N2CC(COC)(NC(=O)CC(C)NC(N)=O)C2)=O)CC2CCC1CC2 45061,C1(O)(C(N(C)CC2CCCCC2NC(=O)Cc2nncs2)=O)CCCC(C)(C)C1 45062,C1(COC)(CONC(C2CC3CC3C2)=O)CCCO1 45063,C(C)(CCCC(=O)NC(CO)CCC1CC1)NC(c1n(CC)nnc1)=O 45064,Cc1ccc(CN(C2CCCCC2)C(=O)NCc2cccc(C(=O)OC)c2)cc1 45065,c1(C(=O)NCCC(C)N(C(C(C)OCCC=C)=O)C)ccc(C(C)C)s1 45066,C1(C2CCN(C(=O)CC3CCSCC3)C2)(NC(c2cc(C)sn2)=O)CC1 45067,C1(N(C(c2ccc(CC)[nH]2)=O)C)CCCC2CN(C(C3(F)CCCCC3)=O)CC12 45068,CN1CCC(F)(F)C(CNC23C(NC(=O)OC(C)(C)C)C4CC2C3C4)C1 45069,C1(C(=O)NCCN(C(C2C3CCC23)=O)CC)CCC(C)=C(C)C1 45070,CC(CCNC(=O)CCCCNC(=O)C(C)n1cccn1)CCO 45071,C=CCC(C(=O)NC(C)CCNC(c1cc2ncccc2s1)=O)C(C)C 45072,C1(NC(CC(C)CF)=O)CCCC12CCN(C(c1cnn[nH]1)=O)CC2 45073,N1(C(C2C(C(C)(C)O)C2)=O)CCC(O)(CCNC(C23CCC(C)(C2)OC3)=O)CC1 45074,c1(NC(C2CN(C(c3nccnc3Cl)=O)CCN2)=O)nc2c(s1)COCC2 45075,CC1CN(C(c2c(F)cncc2Br)=O)CC2(CCN(C(=O)CO)C2)O1 45076,Cc1ccc(CCC(=O)NC2CC(CNC(c3cnnc(O)c3)=O)C2)cn1 45077,C(=O)(C#CC1CCCCC1)N1CCC(NC(C(C)N(CC(F)(F)F)C)=O)C(O)C1 45078,Cc1cc(CC(=O)NCC23CC(CNC(=O)C(C(C)C)N(C)C)(C2)C3)cc(F)c1 45079,CC(C)CC(C)(CNC(C1(C#N)CC(C)C1)=O)NC(c1ccc(NC=O)cc1)=O 45080,N1(C(C2(N(C)C)CC2)=O)CCN(C(c2cccc(CC#N)c2)=O)CC(O)C1 45081,C(=O)(CCCCC(C)C)NC1C2(CNC(c3cncc(C)n3)=O)CCC(C1)C2 45082,N1(C(c2n(C)nnc2)=O)CCCC(C2CC2NC(C2CCCN2S(C)(=O)=O)=O)C1 45083,c1(C(=O)NC2CC(NC(C3(CC)CC3)=O)C2)cc(=N)[nH]cc1Br 45084,C1(CC2N(C(C)=O)CCC2)CCN(C(c2cn(CC(=O)N(C)C)nn2)=O)CC1 45085,c1(C(=O)NC2(CNC(CCOCC)=O)CC2)cccc2nn[nH]c12 45086,c1(OC)ccc(CN2CC(NC(CSc3ccccc3)C(=O)O)C2)c(Br)c1 45087,c1(C(=O)NC23CC(NC(C(c4cccc(C)c4)C)=O)(C2)C3)cc(F)c(N)cc1F 45088,c1(C(=O)OC)cc(NC(c2ccc3c(n2)OCCO3)=O)cc2[nH]ccc12 45089,C1(NC(C2CCC(C)(C)CO2)=O)CC2CCC1CC2NC(=O)CC1CCCOC1 45090,c1(C(=O)NC2CC(CNC(C3CC=CC3)=O)C(O)C2)ccc2oc(O)nc2n1 45091,C=C(C)C1OCCC1C(=O)NC1CN(C(=O)COc2cncc(Cl)n2)CC1OC 45092,c1(C(=O)NCC2(NC(=O)C3=CCCCO3)CCC2)cc(Cl)cc([N+](=O)[O-])c1 45093,C(C(C)(C(=O)N1CC(C(N)=O)C(O)C1)OC)OC.C1CCC(=O)N1C 45094,c1(OC)ncnc(OC)c1CN1CCC(NC(=O)Cn2ccnn2)C1 45095,C1(NC(c2c(C)cccc2F)=O)CC1C1CCN(C(=O)Cc2csc(Cl)c2)CC1 45096,N1(C(C(C)OCCC#C)=O)CCOC(C)(CNC(c2ccc(OC)c(F)c2)=O)C1 45097,C1(C(C)C)N(C(=O)N(Cc2ccccc2)Cc2nc(C(C)O)n[nH]2)CC12CCC2 45098,C(c1cn(C)c2ccccc12)=CC(=O)NC1C(C)CN(C(c2cnn[nH]2)=O)CC1 45099,C1(N(C(=O)Cc2cnoc2)CC)CCCN(C(=O)CC2CC(F)(F)C2)CC1 45100,N1(C(c2nc(Br)cs2)C(=O)NCCCSC)CCC(CCO)CC1 45101,C(=O)(CC(O)CC(C)(C)C)N1CCN(C(CCCCN(C(C)=O)C)=O)C(C)C1 45102,C1(N=c2cncc(Cl)[nH]2)(CNC(=O)CN2CCCC2=O)CCOCC1 45103,O=C1OCCC2CN(c3ncncc3-c3ccccc3)CC12 45104,n1(CCC(=O)N(CCF)CCc2ccccn2)cc(COc2ccccc2)nn1 45105,CCCCC(C(=O)NCc1ccnc(O)c1)NC(=O)CC1CC2CC2C1 45106,C1(CNC(C(C2CN(C(C(C(=O)OCC)F)=O)C2)O)=O)OC(=O)NC1(C)C 45107,CC(C)CCC=CC(=O)NC(C)C(=O)NCC(C1CC1)N(C)C 45108,N1(C(C(C)OCCN(C)C)=O)CCC(NC(c2cncc(N)c2)=O)CC1 45109,N1(C(C(C)O)=O)C2CCC1CN(C(=O)CCCCC(N)=O)C2 45110,N1(C(C2(C)CC(C)(C)C2)=O)CCC2(CCC(CNC(C3CC3(C)C)=O)OC2)CC1 45111,Cc1cccc(Cl)c1OCC(=O)NC1CN(C(C2CC(C)(F)C2)=O)CC12CC2 45112,n1(CC(=O)Nc2cc(Cl)on2)cc(CNc2ccncc2)nn1 45113,Cc1cc(F)ncc1C(N1CCN(C(=O)CCCCCF)CC1C)=O 45114,N1(C(c2ccc(N(CCC)C)nc2)=O)CC(C)(C)CC1CNC(=O)C(C)N(C)C 45115,NS(=O)(=O)CCN=c1[nH]c(N(C)Cc2ccc(Br)s2)nc2c1CCC2 45116,c1(CN2CC(F)(C(=O)Nc3cc(CC)cc(Br)c3)C2)cc(Cl)c(O)cc1F 45117,N1(C(C(C)=C(CC)C)=O)CCN(C(C2(S(C)(=O)=O)CCC2)=O)CC1CC(=O)NC 45118,CC1(c2cn(C3CCCN(C(=O)C(C)(O)C(F)(F)F)C3)nn2)CCC(F)(F)CC1 45119,CC1CCN(C(=O)CC2C=CCCC2)C1C(=O)N(C)CCC1CCCC1 45120,C1(NC(c2ccc(OC)cc2)=O)CCC(C)N(C(c2ccc(F)c(Br)c2)=O)C1 45121,N1(CC#N)CCCC1C1CCCCN1C(c1cccc2nc(O)[nH]c12)=O 45122,C(CC1CCC1)(C(=O)N(C)CC1CCN(C(c2cc(C(C)(C)C)no2)=O)C1)OC 45123,c1(N2CCC(CC=C)(NC(c3cc(C4(C)CC4)n[nH]3)=O)C2)ncnc(Cl)c1CO 45124,C1(CNC(c2n(C)c(S)nc2)=O)CC2(CCN(C(C3CCCC3O)=O)C2)CO1 45125,N1(C(CCN(CC(C)(C)C)C2CC2)=O)CC(CO)C2(CCNCC2)C1 45126,c1(NC(C2CCC2F)=O)cc(C(F)(F)F)c(Cl)cc1F 45127,C1(NC(c2c(OC)ccs2)=O)CC2CC(NC(=O)CCC(C)CN(C)C)C1C2 45128,N1(C(c2c(OC)nccc2)=O)C2CCC1C(C(=O)Nc1ncccc1C(C)C)C2 45129,c1(C(=O)NC2CN(C(c3n(CC)nnc3)=O)C(CO)C2)ccc2nnn(O)c2c1 45130,C(=O)(C1=CS(=O)CCC1)N1CC=CC(NC(CCc2cn(C)nn2)=O)C1 45131,Cc1nn(C)c(-n2cccn2)c1C(=O)NC1CCCN(c2ccccc2F)C1 45132,N1(C(C2CC(N(C(CC3(N(C)C)CC3)=O)C)C2)=O)CC2(CCC2(C)C)C1 45133,C1(CN(C(=O)CCn2cnnn2)C)CN(C(c2cccc(O)n2)=O)CC12CC2 45134,c1(CCC(N2CCN(C(C(CC)O)=O)CC2C(C)C)=O)ccc(S(C)(=O)=O)cc1 45135,N1(C(C2(C(=O)OC)CC2C)=O)CCC2(CCCN2C(C2CCCC2C)=O)C1 45136,c1(N2CC(C)(CNC(CCC)=O)OCC2)cc(C)c([N+](=O)[O-])cc1F 45137,C(CC(=O)NCCC1=CCCCC1)(C(C)C)NC(C(C1CC1)OCC)=O 45138,c1(C(=O)NCCC(C)(C)NC(C2CC23CCCOC3)=O)c(Cl)ccc(F)c1F 45139,CCCC(C)CCCC(=O)NC1CCC(C)N(C(=O)C=Cc2ncc[nH]2)C1 45140,C(=O)(C#CC1CCCOC1)N1C(C2(NC(Cc3ncc(C)s3)=O)CC2)CCCC1 45141,C1(C(=O)NC2CN(c3nccc4c(Br)csc34)C2)CC2(CO1)CC1(C2)OCCO1 45142,N1(C(c2cncc(NC(CC)=O)c2)=O)CC2(CCC(NC(c3ccoc3)=O)C2)C1 45143,N1(C(CNC(=O)OCC)=O)CCCC2(NC(=O)Cc3ncccc3C)CC12 45144,S(=O)(=O)(c1cccc(CBr)c1)N1CCC2CN(C(c3cc(Br)nc(Br)c3)=O)CC21 45145,C1(N(C(c2c(COC)cco2)=O)C)CCC(NC(C2CC3(CC3)CO2)=O)CC1 45146,N1(C(C(C)OCC=C)=O)CCC2(CCCN(Cc3cc(C)ccc3O)C2)C1 45147,CC1CN(C(=O)CC2OCCC2(C)C)CC1NC(=O)Cc1n[nH]c(=N)s1 45148,c1(CC(N2C(C)CC(NC(C3CCC(C)C3)=O)C2)=O)ccc2sccc2c1 45149,c1(C(C)C)nc(C(=O)N(C2CN(C(=O)C(C)CN3CCCCC3)C2)C)cs1 45150,C1(CNC(CSCCN(CC)CC)=O)CC2(CO1)CN(C(=O)CN(C)C(N)=O)C2 45151,S(=O)(=O)(CCC(F)(F)F)N(c1ncc(C#N)cc1Cl)C1C(C)CCNCC1 45152,N1(C(c2nc(C)c(C)s2)=O)CCN(C(=O)C=CC2CCC2)CC1CC1CC1 45153,C1(NC(c2cc(C)c(O)nc2)=O)C2CC3CN(C(=O)CC(C)(C)C(F)F)C1C3C2 45154,N1(C(c2[nH]cc(C#N)c2)=O)CC2(CCC2)CC1CNC(C1(N2CCCC2)CCC1)=O 45155,N1(C(CSc2c(C)n[nH]c2C)=O)CC2(CCC2)CC1CNC(C1(F)CCOC1)=O 45156,N1(c2nccc(OC)n2)C2CCCC1CN(C(C1(O)CCOC1)=O)CC2 45157,C(C(=O)N(CCCCN(C(=O)CC1C(=O)NN=C1C)C)C)(C(C)C)OCC 45158,C(C(CC)(CC)C(=O)NC(c1ccccc1)C)NC(C(CC=CC)C)=O 45159,c1(N2CC(C(C)NC(C3(C)CC(O)CN3C)=O)C2)ccc([N+](=O)[O-])cn1 45160,N1(C(Cc2cnc(C)[nH]2)=O)CCCC2CN(C(=O)C(C)CS(C)(=O)=O)CCC12 45161,C(C(=O)N1CC(=O)NC(C)C1)(C(C)(C)C)n1cc(C(=O)OC)nn1 45162,C(=O)(CCC(C)(C)NC(C1CCC(=O)C(C)C1)=O)NCCC(CCC)C 45163,c1(CC(=O)N(C2CCN(C(C3CCCN3S(C)(=O)=O)=O)C2)C)ncc(F)cc1F 45164,C(CC(C)C(=O)NCCC1(CNC(C2(C(F)F)CCCC2)=O)CC1)=CCC 45165,C1(CC=C)(NC(=O)C(CN(C)C)NC(=O)Cc2cnn(CC)c2)CCCC1 45166,c1(NCC)ncc(C(N2CC3C(NC(C4CCCCNC4=O)=O)C3C2)=O)cc1Cl 45167,C#CCC(CC(=O)N1CCC1CC(=O)NC)NC(=O)C(C1CCC1)OC 45168,c1(CC(=O)NCc2ccc(-c3ccc(CO)cc3)cc2)nc(Br)n2c1CCCC2 45169,CC1(C)CC(CCNC(C2CCN(C(=O)CS(C)(=O)=O)CC2)=O)CO1 45170,CCCC(CCCNC(=O)C(CC)C(C)C)NC(c1csc(-c2ccco2)n1)=O 45171,CCP1(=O)CCN(c2ccc(NC(=O)OC(C)(C)C)nc2)CC1 45172,c1(CNCC(n2cnc(-c3cccs3)n2)C)cccc(Cl)c1 45173,N1(C(CC(=O)NCC)=O)CC2CN(C(=O)CC(C)C(C)C)CC2(C)C1 45174,C1(CNC(CCC=C=C)=O)CC(C)CN(C(=O)C(C)CCC)C1 45175,C1(C(N2CC(C=C)C(NC(=O)C3=COCCC3)C2)=O)CC12CCCCCC2 45176,C1(CNC(c2ccn(C)c2)=O)CCC(F)(CNC(C2CC3CCC(C2)S3)=O)CC1 45177,c1(OC)ccnc(C(=O)N(CCCCNC(C2CCC(C(F)(F)F)O2)=O)C)c1F 45178,C(=O)(C(C)C(O)C(C)CC)N1CC(C(=O)NCC(CC)N(C)C)C(C)(C)CC1 45179,N1(C(C(CCNC(=O)CC2OCCO2)OC)=O)CCOC(C)(C)C1C 45180,C1(NC(c2nc(C)oc2)=O)CCCCN(C(=O)COCC2CCCC2)CC1 45181,Cc1cc(F)cnc1C(=O)NCC1CN(C(=O)CCn2ccnc2)CC1O 45182,N1(C(COC)=O)CCOC(CNC(=O)CNC(c2ccnc(N(C)C)c2)=O)C1 45183,C(C)(C(O)C(F)F)NC(C=CCN(C(c1cn(C(C)C)nn1)=O)C)=O 45184,CCCCCC(C)(C)C(=O)NC1CN(C(=O)C(C)SC(F)(F)F)CCC1C 45185,C1(C(N2C(CNC(C3N(C)CC4(CC4)C3)=O)CCC2)=O)CCC(C2CC2)CC1 45186,N1(C(C(CC)=CCCC)=O)CC(=O)CC1C(=O)NCc1cc(O)ncn1 45187,c1(C(C(=O)OC)NC(C2NCCCC2C(F)(F)F)=O)ccc(F)c(Cl)c1 45188,CC1(C(N2CCC(F)(CNC(=O)C#CC3CC3)C2)=O)CCC(F)(F)CC1 45189,c1(C(N(CCOCCCNC(c2ccc(OC)s2)=O)C)=O)ccn2cccc2c1 45190,C(=O)(C(C)(C)CN1CCN(c2nc(C(=O)O)cs2)CC1)OC 45191,c1(C(N(C2CCCC(NC(c3c(C)occ3)=O)C2)C)=O)nn(C)c2c1CCC2 45192,c1(C(=O)NC(c2nc[nH]n2)CC)ccoc1CNC(C1CC1(C)CC)=O 45193,N1(C(CC(CCC)(C)O)=O)CCC2C1CCCN2C(c1cn(C2CC2)nn1)=O 45194,c1(CC(=O)NC(C2CCOC2)CNC(C2(F)CC=CC2)=O)ccccc1Br 45195,CC(C(=O)NCC(C)CN(C(=O)COc1ccc(OC)cc1)C)S(N)(=O)=O 45196,c1(C(=O)NCC2(F)COCCN(C(C=NOC)=O)C2)cnc2scc(C)n2c1=O 45197,C(CN=[N+]=[N-])(C(=O)NCCCc1ccccc1)NC(COCC=C)=O 45198,c1(C(=O)NC(C)CNC(=O)C(c2ccc(C#N)cc2)O)cnn2cccc(Cl)c12 45199,C(CC(=O)CCO)c1cn(CCCCN(C(=O)C=CC2CCCC2)CC(=O)O)nn1 45200,c1(CNC(C(CC)O)=O)ccc(CNC(C2CCCC2C(C)C)=O)cc1 45201,c1(C(C(=O)NC(CC)(C)C)N(CCC#N)C2CCC2)ccc(Br)c(F)c1OC 45202,CC1(C)CCCC1C1CCN(c2cc(N3CCOC4(CCC4)C3)ncn2)C1 45203,CC(C(=O)NC(CNC(c1c(F)cncc1Cl)=O)C1CCC1)C(F)(F)C(F)F 45204,N1(C(C)=O)CCC(NC(c2[nH]nc3c2COC3)=O)C(F)C1 45205,CCCCCCCCCCN(C(C1CS(=O)(=O)C1)=O)Cc1nnc(C)n1C 45206,C(C1CCCc2cccnc21)NC(NC(CC)C)=NCCNC(=O)COC 45207,C1(NC(c2cc(OC)ncc2Cl)=O)CN(C(C2CC=CCC2C)=O)CC(F)(F)C1 45208,c1(C(=O)NC2(C)CCN(C(C=C(C)CN3CCOCC3)=O)C2)ccc(N)c(C)c1Cl 45209,CCCCC(O)CNC(C1CCCCN1C(c1ccc(OC)o1)=O)=O 45210,c1(C(N2CC3(CCN3C(=O)CS(=O)C(c3ccccc3)c3ccccc3)C2)=O)cncc2cnccc12 45211,C1(C(N2CC(C(C)(C)C)OCC2)=O)C2CCN(C(n3cc(C4CC4)nn3)=O)CC12 45212,N(C(=NCc1cn(C)nc1OC)NCc1ncnn1C)C(CC)CC 45213,CN1CCN(C(=O)CC2(NC(=O)CC3CC4CC4C3)CC2)CC(O)C1 45214,c1(OC)cc(C(N2CCN(C(=O)COCC3CC3)C(C)C2)=O)c2cnccc2c1 45215,c1(C(=O)NC2CCN(C(C(C)(C)N(S(C)(=O)=O)C)=O)CC2)ccc(CN)cc1O 45216,c1(C(=O)NCC2CN(C(c3ccoc3)=O)C2)ccc(Br)cn1 45217,Cn1cc(C(N)=O)cc1C(=O)NC1CCC1NC(=O)C1=NOCC1 45218,C(C(F)C(=O)N1CC(F)C1)C1CN(C(C2(CC#C)CC2)=O)C1 45219,C1(NC(=O)CC23CCCN2CCC3)CN(C(=O)Cn2cnnc2)CC1C1CC1 45220,N1(C(CN(C(c2cccc(C#N)c2)=O)CC)=O)CC2(CC(F)C2)C1 45221,C(=O)(CCC(C)(C)NC(C1CCC(CO)CC1)=O)N(C)CC1CCC(C)CC1 45222,N1(Cc2cnn(C)c2Cl)CCC(F)(F)C(C(=O)Nc2nc(C(C)C)cc(Cl)n2)C1 45223,c1(OC)cc(C(N2CC(CNC(c3ccsc3OC)=O)C(C)C2)=O)ccc1F 45224,C1(O)(CNC(=O)CCCC2CCCC2)CCCN(C(C2COC(=O)O2)=O)C1 45225,C#CCCC(O)C(=O)NC1(CCC)CCCN(C(=O)Cc2ccnc(O)c2)C1 45226,N1(C(C2(OC)CC2)=O)CCC(CN(C(=O)C=CC(N2CCOCC2)=O)CC)CC1 45227,C(=O)(C(CC1CC1)NC(C1(CCNC(=O)CCc2nc(O)n[nH]2)CCC1)=O)NC 45228,CC1(C)CC(CNC(c2cccnc2)=O)N(C(=O)Cc2cncnc2)C1 45229,c1(C(=O)NC2C(NC(C3C(C#N)CC3)=O)C2)ccc(C2CCCCC2)cc1 45230,c1(C(=O)OC)ccc(C(=O)NCCCCNC(c2nc(=O)n(C)[nH]2)=O)nc1 45231,C(=O)(C(C(C)NC(=O)CCCN(C)C)C(C)C)N(CC#C)C1CC1 45232,Cc1c(CC(N2CCC(CCCO)C2)=O)c(=O)oc2cc(N)ccc12 45233,Cc1cc(C(N2CC3CC(C2)C3NC(C2CCNC(=O)C2)=O)=O)n2nccc2n1 45234,C=CC1CN(C(C23CCOC(C)(C2)C3)=O)CC1NC(c1csc(F)c1)=O 45235,CCC(CC(=O)NCC1CN(C(=O)CC(C)(F)F)CC1C(F)(F)F)C(F)F 45236,c1(CC(=O)NCC(CC=C)NC(C2CC(C)=NO2)=O)ccc(Br)c(Cl)c1 45237,C1(CNC(C2=CC(C)(C)C2)=O)CC2COCC2N1C(=O)COc1ccccn1 45238,N1(C(C(=O)NCC(F)F)c2ccsc2)Cc2nccc(Cl)c2C1 45239,c1(CC(C(=O)NC(CCCNC(c2occ(C)c2)=O)C)C)c(C)n[nH]c1C 45240,c1(C(=O)NCC(C)NC(CCn2ncc(C)c2)=O)ccc(Cl)cn1 45241,c1(CC)ccc(C(=O)NCC(C)(C(C)C)NC(=O)CCc2cnc(O)[nH]2)cn1 45242,C1(C(N(C2CCN(C(c3csc(=N)[nH]3)=O)C2)CC#C)=O)CC(C)(C)CCO1 45243,C1(NC(C(CCC)O)=O)CCN(C(c2cocn2)=O)CC12CCC2 45244,Cc1cc(-c2nc(C)c(C(=O)N(C)CCN(C(=O)CCC(C)C)C)s2)ccc1F 45245,c1(C(N(C2CCCN(C(CCCC#C)=O)C2)CC)=O)ccc(C)c(Cl)c1 45246,CC#CCC(C(=O)Nc1cncc(C(N)=O)c1)NC(C1CCCCC1O)=O 45247,c1(C(=O)NC2CC(CNC(C(C)CC(C)(C)C)=O)C2)ccc2c(c1)CCCC2 45248,C1(C)(CNC(C(C(C)C)NC(N)=O)=O)COCCN(C(=O)C2=CCCCO2)C1 45249,C1(CNC(c2cc(SC)oc2)=O)CC12CCN(C(=O)C(O)CC(F)(F)F)CC2 45250,c1(CNC(C2(C)CCN(C(c3cscn3)=O)C2)=O)cc(Br)ccc1Cl 45251,CC(O)C(C)C(=O)NC(C1CCCN1C(=O)CSCC(N)=O)(C)C 45252,c1(C(=O)NC(c2cccc(C)c2)CNC(C=COC)=O)nn2c(c1C)CCCC2 45253,Cc1cc(C(N2CCC(O)(C(C)NC(C3CC(F)C3)=O)C2)=O)ncc1C(F)F 45254,C(c1ccc(F)cc1[N+](=O)[O-])=CC(=O)OCCc1c[nH]c(=N)s1 45255,c1(COC)ncc(C(=O)NC2CC(NC(=O)Cn3cc(C)ccc3=O)C2)c(O)n1 45256,C=CC1CCCCN1C(C1CC=CCC1NC(c1ncn(C)c1C)=O)=O 45257,C(=O)(C(F)C(C)(C)O)N1CC(CCC=C)(C(=O)Nc2c[nH]ccc2=O)C1 45258,c1(NC(c2n(CCCSC)nnn2)c2csc(Br)c2)cc(O)c(C)cc1C 45259,N1(CC(=O)NC(CNC(c2cc(C3(C)CC3)n[nH]2)=O)(C)C)CCS(=O)(=O)CC1 45260,c1(SC)ccc(C(=O)NCC(C)(C2CC2)NC(=O)COCC(=O)CO)cc1 45261,c1(C(=O)OC)cc(CNC(C2CSCCN2c2ccnc(C)n2)=O)cc(CO)c1 45262,N1(C(CNC(CC)=O)=O)CCCOC(CNC(c2ccc(C)cc2C)=O)C1 45263,c1(C(=O)NCc2c(CN(C(CC)=O)C)cccc2)cc(C#N)c(N)cc1O 45264,C(=O)(C(C)CC(C)C)NCC(CNC(c1cc[nH]c1)=O)OC 45265,c1(C(=O)NC(CN(C)C)C(=O)NCC(O)CC(F)(F)F)cc(F)cc(F)c1 45266,c1(C(=O)NCC(CNC(C=CC(=O)OCCCC)=O)O)nn[nH]c1Cl 45267,C#Cc1ccc(F)cc1C(N1CCOC(CN(C)C(c2ccc(SC)s2)=O)C1)=O 45268,c1(C(=O)NCCN(C)C(C2(CS(C)(=O)=O)CC2)=O)cccc(CC2CC2)c1 45269,CC1CCC(C)C(C)C1NCC1CCC(=O)N1 45270,C1(CCN(C(c2cnc(C(C)C)s2)=O)C)CCCCN1C(=O)C(C)C1(O)CCC1 45271,C(CC(C(=O)NCC1CCN(C(C)C)C1)NC(c1sccc1C)=O)OC 45272,c1(C(N2CC(OCCNC(=O)C(F)CC3CCCC3)C2)=O)ccc2sncc2c1 45273,C12(COC)CNC(C(N3CCN(C4CCCC4O)CC3)=O)(C1)C2 45274,c1(CNC(c2ccc(OCC(=O)N(C)C)cc2)CC(C)C)ccc2c(c1)OCO2 45275,c1(C(N2CC(C)(C(=O)Nc3ccnc(F)c3)C2)=O)c(F)c(F)cc(F)c1F 45276,Cc1cc(C#N)nc(N2CC(C)CC2C(N2CCC(OC(F)(F)F)CC2)=O)n1 45277,CC(C)(C(F)(F)F)OCC(=O)NCCOCCNC(C1(F)CC=CCC1)=O 45278,c1(C(N2CCC(CNC(C=CCOC)=O)(OC)CC2)=O)ccc(C)c(C)c1O 45279,N1(c2nnc(C)s2)CC(CNC(C2(C)CC(C)(C)C2)=O)OC2(CCC2)C1 45280,C1(CC)C2CN(C(c3ccc(C)s3)C(=O)NC)CC12.C1(=O)CC(C)N1 45281,c1(CC(=O)NC(C)CCNC(=O)C(C)n2cncn2)cc(F)cc(Cl)c1 45282,C1(C(=O)NCCN(CCOC)C(c2nc(Cl)cs2)=O)CCCC1OC 45283,Cc1noc(C(F)(F)F)c1C(=O)NCC(F)CNC(C1(C2CC2)CC1)=O 45284,c1(CCC(N2C(CNC(c3ccc(COC)[nH]3)=O)CC2)=O)ccc(SC)cc1 45285,c1(N2CC(CC)OCC2)cc(Br)ccc1S(=O)(=O)N(C(C)(C)COC)C 45286,C(=O)(C1COc2ccccc21)N1CC(CCNC(c2cc(C)n(C)c2)=O)OCC1 45287,Cc1cc(CC(=O)NCCCCNC(=O)CCC(=O)c2ccncc2)c(C)s1 45288,N1(C(c2c(C)nn[nH]2)=O)CCN(C2CCCN(C(=O)C(C(C)C)N(C)C)C2)CC1 45289,C1(C(=O)NC(C#C)CCC)CC(=O)CN1C(C1(C(=O)C2CC2)CC1)=O 45290,N1(C(c2c(C3C(C)C3)noc2)=O)CCC(C(=O)NCCNC(C2CCC2)=O)CC1 45291,n1(CC)ccc(=NC(=O)C2CN(C(c3ccccc3O)=O)CCC2(C)C)[nH]1 45292,N1(C(CCC2C(C)C2)=O)CCN(C(C2(NC(N)=O)CCCCC2)=O)CC1CCO 45293,C1(CNC(C2C=CCN2C(=O)C(O)C2CCCC2)=O)CC2(CCC2)C1 45294,c1(C(c2n(CC=C)nnn2)NCc2ccns2)ccc(C)cn1 45295,N1(C(Cc2ccc(C)s2)=O)CCCC(N(C)C(C2C(C)OC(C)C2C)=O)CC1 45296,C1(C(=O)NCC(C)C(=O)NC2C=CC(C)(C)CC2)CCC(C)(O)CC1 45297,c1(C(C)C)ccc(OCC(N2CC(NC(=O)Cc3csc(Br)n3)C2)=O)cc1 45298,CC(CS(C)=O)C(=O)N(CCCNC(=O)CNC(=O)CCCCO)C 45299,C(C(C)(C(=O)NCC=CCC(=O)NCC(C)(C)O)OC)OC 45300,C(=O)(C1=C(Cl)CCOC1)NC(C(C)(C1CCC1)NC=O)=O.c1(C)cccnc1O 45301,C(=O)(CS(=O)(=O)c1nccn1-c1ccccc1)N1C(c2n(CC)ncc2)CCC1 45302,c1(NC)cnc(Cl)cc1C(=O)NCC1CCC(NC(C2COCCO2)=O)C1 45303,c1(C(=O)OC)cc(Cl)c(OC)cc1C(C)C.c12ncc(s1)CNC2 45304,C#CC(C(C)(C)C)NC(=O)C(C)(CSC)NC(C1SCC=C1C)=O 45305,c1(-c2cn(C)nc2)ccc(F)c(NC(=O)NCc2cn(CC3CCCC3)nn2)c1 45306,c1(C(c2nnnn2CC2CCOC2)NCc2ccn(C)n2)c(Cl)cncc1Br.C1CC1 45307,n1(CCCC)ncc(C(=O)NCC(O)CN(C)C(c2nnn(C)c2C)=O)c1CC 45308,N1(C(C)=O)CCCC1C(=O)NC(C)(CNC(c1cn(CC(N)=O)nn1)=O)CO 45309,C1(CNC(C(c2cnn(C)c2)C)=O)CCC(NC(=O)Cn2cncn2)CC1 45310,C(=O)(C1=CCCC1C)NC(CCOCC)C(=O)NCCNC(c1ccoc1)=O 45311,C1(C(N2C(CN(C(CCCOCC=C)=O)C)CC(F)C2)=O)CC(C)CC(C)(C)C1 45312,Cc1ncccc1C(N1CC=CC1CNC(C1C(F)(F)C12CC2)=O)=O 45313,c1(OC)ccnc(-c2cn(C3CCN(C(C4(C)C=CCCC4)=O)C3)nn2)c1 45314,c1(C(=O)NCC2(O)CN(C(CSc3n(C)nnn3)=O)C2)cnc2n1CCC2 45315,c1(OC)cccc2c1OCCCC2NC(=O)C(=O)NC1CCN(C(C)C)C1=O 45316,N1(C(c2c(CC)cco2)=O)CCC(C2CC2)C1C(N1CC(CO)C2(CC2)C1)=O 45317,N1(C(CCCNC(=O)C(C)OC2COC2)=O)CCCOC(CSC)C1 45318,CC1(C(=O)NC2CC(CNC(C3(C(F)F)CCCC3)=O)C2)CCCNC1=O 45319,c1(CN(C(C2CCCSC2)C(=O)NCC)C2CC2)c(C)nn(C)c1C 45320,C1(NC(=O)CC2CCC(O)C2)CC2CCC(C1F)N2C(c1nc(Cl)c(Cl)s1)=O 45321,C1(C(N2CCN(C(c3cccc(O)c3)=O)CC2)=O)(OC)CC(C)CC(C)C1 45322,CC1CCC(NC(=O)NC2CN(CC(F)(F)F)C2)C(C)C1 45323,N#CC1CC(C(=O)NCC(O)CNC(C2(CC3CCC3)CC2)=O)C1 45324,C12(C=O)CC(CN(N3CC(C(CC)CC)C3)C1)C2.n1(C(C=O)C)ccnc1C 45325,CCCC(C)CC(=O)N1CCOC(CN(C(=O)COC2CC2)C)C1 45326,N(C(=NCCC)NCCC(C)Oc1cccc(C(F)(F)F)c1)CC=C 45327,N1(C(C2(CC#C)CC2)=O)CC(C(N2CCOCC(=C)C2)=O)C(F)(F)C1 45328,N(C1CN(c2cc(Cl)ncn2)CCc2ccccc21)C(=O)CCc1cnc[nH]1 45329,C1(C(N2C(C)CC(CNC(c3cc(O)nn3C)=O)C2)=O)CCn2c(O)nnc2C1 45330,C12(CNC(c3c(CC)nc(=N)[nH]c3)=O)CCCC(CN1C(c1cnsc1)=O)C2 45331,c1(C(=O)NC2CCN(Cc3c(C#C)cccc3)CC2O)ccc(O)c(O)c1Cl 45332,c1(COC(=O)CNC2CCN(C(c3cnoc3)=O)CC2)ccc2nccn2c1 45333,c1(COC)nc(NCC2CC2C2CCC2)cc(=NCCSC2CCCC2)[nH]1 45334,c1(C(N(CCCNC(C2C(=C)C2)=O)C2CC2)=O)ccc(OC)c(S(N)(=O)=O)c1 45335,N1(C(C(C(C)C)NS(C)(=O)=O)=O)CCC(C)CC1CNC(=O)CN(C)C(C)C 45336,c1(OC)ccccc1C(N1CC(N(C(=O)CCC(C)N(C)C)C)C(O)C1)=O 45337,Cc1[nH]c2c(C(N3CCC(CNC(=O)CC4CC4(Cl)Cl)C3)=O)cccc2c1C 45338,N1(C(C(C(C)(C)O)F)=O)CCC(C2(NC(c3cc(C4CC4)nnc3O)=O)CC2)C1 45339,c1(CN2C(C(=O)NCC(O)CO)CC(O)C2)cc(Br)ccc1F 45340,N1(c2c(OC)cnc(Cl)n2)CCCC(C2CC2NC(=O)Cc2occc2C)C1 45341,c1cc(C)cc(C)c1Br.c1(C(=O)OC)cccc(O)c1F.c12cn(nn1)C2 45342,C1(O)(CCNC(c2c(C)nc(CCC)s2)=O)CCN(C(=O)C(CC)OCC)CC1 45343,N1(C(c2c(C)nc(C(C)C)s2)=O)CCN(C(=O)CSc2nc[nH]n2)C(CO)C1 45344,Cc1cc(N2CC(C)(C)CC2CNC(c2csc(CO)n2)=O)nc(C)n1 45345,c1(C(=O)NC2(C3CC3)CCN(C(C(CC)(C)C#N)=O)C2)cnc2ccncc2c1 45346,C(=O)C1=CCCNC1.c1(C(NOCCCC)=O)[nH]ccc(=O)c1C 45347,c1(C(=O)NC(C(C)NC(C2CC(=C)C2)=O)(C)C)cc(Cl)cc(F)c1N 45348,c1(C(=O)NCCN(CCC)C(C2CCCSC2C)=O)occ2c1CCC2 45349,C1(NC(c2ccccc2Cl)(C)CO)CC2CCC(C1)C2N 45350,c1(C(=O)NC2(COC)CN(C(c3n(CC)c(O)nc3)=O)C2)cncc([N+](=O)[O-])c1 45351,C#CC1(NC(=O)C(C2(C)CC2)NC(=O)C(CC)CC=CC)CCCCC1 45352,N1(C(CCc2cc(C)on2)=O)CC(C)(C)CCC1CNC(C1CCCNC1=O)=O 45353,N1(C(CCN(CC#C)C(c2cccc(C#C)c2)=O)=O)CC(C)(COC)CC1(C)C 45354,CC(C)CCC(C)NC(=O)CN(C(=O)CC1CC2(CC2)C1)C1CC1 45355,c1(C(=O)NCC(CN(C)C(C2CCCC2)=O)O)ccc2cnnc(O)c2c1 45356,C(C1CCOCC1)=CC(N1CC(COC)(CNC(C2(C)CCOC2)=O)C1)=O 45357,c1(C(N2C(CNC(C=C(COC)C)=O)CC(F)C2)=O)cccc(OC)c1C 45358,c1(C(=O)NC(C)(CNC(=O)C(O)CN2CCCC2)CO)csc2nnsc12 45359,N1(C(COC)=O)CC(C)(C)CCC1CNC(=O)CC(O)c1ccccc1 45360,N1(C(c2nnn(C(C)(C)C)n2)=O)CC(NC(c2ncccc2O)=O)CC(F)C1 45361,c1(C(N(C(C)CNC(c2ccnn2C(F)F)=O)C)=O)oc2ccccc2c1Cl 45362,C1(F)(CNC(COCCCOC)=O)CCCN(C(C2CCC=CCCC2)=O)C1 45363,C(CC(C(=O)NCCc1nncn1CC)NC(c1cnco1)=O)=CC 45364,N1(C(Cc2nc(C)oc2)=O)CCCC1(C)C(=O)NCC1(C)CCCC1O 45365,c1(OC)ccc(C(=O)NC2CCC2NC(C2CC2c2ccc(F)cc2)=O)c(F)n1 45366,Cc1ccc(F)c(C(CO)NC(=O)C(c2ccc(F)cc2)C2CC2)c1 45367,C1(NC(C(C)OCC#C)=O)CN(C(=O)CCc2cccs2)CC2(CCC2)C1 45368,c1(C(N(CCNC(CCOCC#C)=O)CC2CC2)=O)ccnn1C1CCOCC1 45369,CC1CC(NC(=O)CCCNC(N)=O)CCN1C(=O)CSC(F)F 45370,C(N=c1nc(C(F)(F)F)[nH]s1)C1CC(NC(C2CC(=O)N2)=O)C1 45371,N1(C(=O)Nc2ccc(C)c(C)c2)CC2C(C1C(N1C=CC[SH]=NC1)=O)C2(C)C 45372,N1(C(C(CCN(C)C)O)=O)CC=C(CC(=O)NC(C)(C)C(=O)N(C)C)CC1 45373,CC1(C)CCC=C1C(=O)NC1CN(C(=O)CC2CCCC(=O)N2)CC12CC2 45374,C(=O)(CC(C=C)CCC)NC1CCN(C(c2cn(CC=C)nn2)=O)C12CC2 45375,N1(C(CCCC(C)C)=O)CC2(C1)SCCC2NC(c1ccc(Cl)cc1)=O 45376,C(=O)(C1=CC2(CCOC2)C1)N(C1CN(C(c2nn[nH]c2Cl)=O)CC1O)C 45377,C(=O)(C(C)CC(=O)OC1CC1)N.C1(OCCSC)CCN(C(=O)CCO)C1 45378,C1(NC(=O)CCc2cncs2)CC12CCN(C(C1CCCOC1)=O)C2 45379,Cc1nn(CC(=O)NCC(C)NC(c2ncc(Br)cc2F)=O)c(=O)n1C 45380,N1(C(c2c(=N)cc[nH]c2)=O)C2CCC1CC(CNC(c1ccc([N+](=O)[O-])s1)=O)C2 45381,N1(C(C2N(C(C)=O)CC(O)C2)=O)CC(NC(c2ccnnc2)=O)C(C)(C)C1 45382,c1(C(C(=O)N2CC(CCNC(c3[nH]ccc3C)=O)C2)OC)c(F)cccc1F 45383,N1(C(c2cc(OC)cc(OC)c2)=O)CCCC(C2CC2NC(=O)C(F)C(C)C)C1 45384,c1(C(N(C2CCN(C(C34CCCC3C4(F)F)=O)C2)CC)=O)cnn2cc[nH]c12 45385,C1(C(N(C(C=C)C)C)=O)CCC(CNC(=O)Cc2ccn(CC)n2)C1 45386,c1(CC(N2CCC(NC(C3C(CC)CCC3)=O)C23CC3)=O)n[nH]c2ccccc12 45387,C#CC(CC1CCC1)N(C(=O)CC=CCC)C.C1(=O)CC2(CC2)N1 45388,C1(CS(=O)(=O)NCC2CC(C)(C)OC2)CCCC2(CCOC2)O1 45389,Cc1nc(CN(C(=O)CC2(NC(=O)C(C)C3CC3)CC2)C)n[nH]1 45390,C(=O)(C(CO)C(F)(F)F)N(C1CN(C(c2cc3cc[nH]c3cn2)=O)CC1F)C 45391,C1(C)(COCC(=O)NCC(C)CN(C(=O)CC2CCCC2)C)CCC(=O)N1 45392,C1(C(=O)NC(C2CN(C(C(C)(C)OC(C)=O)=O)C2)C)CC1C1CCCC1 45393,c1(C(=O)NC(CC)CNC(C2(Cl)CC2(F)F)=O)cccc(-c2cscn2)c1 45394,C1(CNC(CC2CCCN(C)C2)=O)CN(C(c2cn(C)nn2)=O)C(C)(C)C1 45395,CCC(C)C(O)C(=O)NCCCNC(c1onc(C)c1C)=O 45396,C(=O)(C(CC(F)(F)F)c1ccc(F)cc1)NCc1nc(Cl)c(C)n1C 45397,c1(CC)[nH]nc(C(N2CC(OCCNC(c3cccnc3C(F)F)=O)C2)=O)c1Cl 45398,N1(C(CCc2n(C)ccc2)=O)CC2CCN(C(c3ncc(F)cc3F)=O)C2C1 45399,C(=O)(C(O)CC(F)F)NC1(CNC(c2c(OC)n[nH]c2)=O)CCCC1 45400,CC1(C)CN(C(=O)CCCC(F)(F)F)C(CNC(=O)CCn2cccc2)CO1 45401,CC1CC(NC(c2ccn(C3CCCC3)n2)=O)CN1C(=O)CN1CC2CC2C1 45402,c1(C(=O)OC)cc(C(=O)NCC(CNC(c2cc(Cl)c[nH]2)=O)CO)no1 45403,C(=O)(C(C)(O)CCc1ccccc1)NC1CC(NC(C(CC=CC)C)=O)C1 45404,C1(C(=O)NCCC(CNC(CN2CC(C)C2)=O)O)CCCN1C=O 45405,C1(NC(C=CCOC)=O)CN(C(c2ccncc2C(F)(F)F)=O)CC(C)(C)C1 45406,CC1CCC(NC(=O)C(=O)C=Cc2ccc(F)cc2)CN1C(C1CCCSC1)=O 45407,c1(OCC(=O)NC(CNC(C(=CC2CCCC2)C)=O)CO)ccc(F)cc1 45408,N12CCCCC(C1)CCC2=O.N1(C(Cc2n(C)ccn2)=O)CCOC(C(N)=O)C1 45409,N1(C(C=C)=O)CCCC2CN(C(c3ccc4cnccc4n3)=O)CC12 45410,C1(NC(C2(C=C)CCOCC2)=O)C2CCN(C(C3(C#N)CCC3)=O)CCC12 45411,CC(C)(C)C(C(=O)NCC1CN(C(=O)CSc2ccccc2)C1)C1CCCCC1 45412,C1(C(=O)NC(C2(O)CCCCC2)C(N2CC(C)(CC=C)C2)=O)CC(C(C)C)=NO1 45413,C1(N(C(c2c(COC)cco2)=O)C)CCCN(C(C2CCCOC2)=O)C1 45414,c1(C(C)(C)C)cc(C(=O)NC2CCCC(NC(C3(C)CC=CCC3)=O)C2)ccn1 45415,C1(CNC(=O)Cc2ccsn2)CCN(C(c2ccnn2C2CCCC2)=O)CC1O 45416,C1(C(=O)NC(C(=O)NCC(C2CC2)OC)C2(C)CC2)CC12CCCCC2 45417,N1(C(CN(C2CC2)CC)=O)CCCC1CC(=O)NCC1(C)CCCS1 45418,C1(C(N(C(CC)CC)C)=O)CCN(C(=O)CC2CNC(=O)O2)C12CCC2 45419,CCCCC(CNC(=O)CCCc1sccc1C)NC(C1(C)CC1(F)F)=O 45420,c1(C(N2C(CCCNC(c3c(OC)ccs3)=O)CCC2)=O)cccc2c1CCO2 45421,c1(C(=O)NC2CN(C(c3c(C)sc(Cl)n3)=O)CC2C)ccc2cnoc2c1 45422,c1(OC)cc(-c2cc(CCC(c3cc(F)cc(F)c3)NC(C)=O)no2)ccc1F 45423,C(=O)(C(C)(C)c1ccn(C)n1)NC(c1ncnn1C)C.C(=O)N 45424,Cc1nc2cc(C(N3CCCN(C(c4ccc[nH]4)=O)C(C)C3)=O)ccc2o1 45425,C1(CC#C)CCCCN1C(=O)NC(c1cccnc1)C1CCNC1 45426,N(C1CCSc2ccccc21)C(C12C(NC(=O)OC(C)(C)C)C3CCC1C2C3)=O 45427,CC1CN(C(=O)CC2C3CCC(C3)N2C(=O)C(C)OC(C)(C)C)C(C)C(C)(C)O1 45428,c1(C(N2CC=C(CNC(Cn3c(C)nc(C)n3)=O)CC2)=O)cnc2c(c1)COC2 45429,c1(CC(=O)NC(CNC(CCCC)=O)CCOC)ccc(OC)cc1F 45430,N1(C(c2c(CC)ccs2)=O)CCN(C)C(C(=O)NCCc2ccccn2)C1 45431,C1(COC)(CNC(c2ccc(O)nc2)=O)CCN(C(C2CCC3(CC3)C2)=O)C1 45432,C(=O)(C(C(=O)OC(C)(C)C)C(C)(C)C)NC1C(CNC(Cn2nnc(C)n2)=O)C1 45433,c1(SCC)ccc(C(N2CC3CC2C3NC(=O)Cc2ccccc2OC)=O)cn1 45434,Cn1cc(C(=O)NCCC2CCN(C(=O)CCCC#N)C2)c(=O)c(Br)c1 45435,NS(=O)(=O)c1ccc(F)c(C(N2CC3(C(=O)NCCC(F)(F)F)CC2CO3)=O)c1 45436,CCC(C)CN=c1[nH]c2c(c(=NCc3ccc4nncn4c3)[nH]1)CCCCCC2 45437,N1(C(C(C)SCC)=O)CCCN(C(=O)C=C(C2CC2)C2CC2)CC1C 45438,C(=O)(CC(Cc1ccccc1)CC)NCCC(=C)CNC(c1cnc(C)[nH]1)=O 45439,C(C(C)(CCO)NC(=O)NC(C1CCOCC1)Cc1nn[nH]n1)OC 45440,c1(C(=O)NC(C2CCN(C(C(CC(C)C)OC)=O)C2)C)ccc(F)c(F)c1F 45441,N1(C(=O)OC(C)(C)C)CC2CCC2(NC2CC(NC(=O)C(Cl)=CCl)C2)C1 45442,N1(C(C2C(C)(CC)C2)=O)CCC(=CCNC(=O)Cc2cccc(C(F)F)c2)CC1 45443,C1(N)CN(C(=O)C2CC2)C1.C12(COC1)C(=O)N(CC)CC2C1CC1.OC 45444,N1(C(CC(C)(C)C)=O)Cc2cccc(CNC(=O)CC3CCCCC(=O)N3)c2C1 45445,c1(CCC(N2CC(NC(c3c(OC)ccs3)=O)C2)=O)cccc2ccccc12 45446,S(=O)(=O)(c1cccc(C(=O)NC2CCC2CNC(=O)C(F)=CCC)c1)NCC=C 45447,N1(C(c2nc(Cl)cs2)=O)CCOC2(CCN(C(C3CCn4nncc4C3)=O)C2)C1 45448,Cc1ccc2cc(C(=O)NC(C)CC3CN(C(=O)C(C#N)C(C)C)C3)[nH]c2c1 45449,c1(C(=O)NCCCC(=O)OC)ncccc1NC(C1C(C(NC2=NCCS2)=O)C1)=O 45450,C1(C(N2CCC(N3CC(O)C3)C2)=O)CCC(Nc2c(C(=O)OC)csc2)CC1 45451,N1(C(c2cc(OC)c(Br)cc2)C(=O)NCCC2CC2)CCC12CCS(=O)(=O)CC2 45452,N1(C(C2(F)CCN(C(c3nc(CC)sc3)=O)C2)=O)CCC2C(O)C(C)(C)C12 45453,C(C)(N=c1ccnc(N2CCCC(c3nncn3CC)C2)[nH]1)c1n(CC)ccn1 45454,Cn1ncc(C(=O)NCC(O)CC(=O)NC2CC2C(C)(C)C)cc1=O 45455,N1(C(CCN(C(CC(C=C)C)=O)CC2CC2)=O)CC2(C1)OC(=O)NC2C 45456,C1(C)(CC)CCCN(C(C2C3CC2N(C(C2CC(=C4CCC4)C2)=O)C3)=O)C1 45457,N1(C(c2ccc(C=CC(=O)OC)o2)=O)CC2OCCN(C(=O)C3CC3)C2C1 45458,CC1CCN(C(C(N2CC(NC(=O)CSC(F)F)C3CC23)=O)C(C)C)CC1 45459,C1(NC(c2ncn(C(C)C)n2)=O)C2CC3C1C3C2C(=O)NCC1CCOC1C 45460,C(=O)(C1=C(Cl)CCC1)N1CC(CN(C(C(CC)(C)C)=O)C)OCC1 45461,c1(OC)cc(C)sc1C(=O)NC1CC(CCNC(C2CCC(C(N)=O)CC2)=O)C1 45462,c1(NC)cc(C(N2CC(c3ocnc3CNC(c3cc(Cl)ns3)=O)C2)=O)n(C)n1 45463,C1(C)(CC)C=C(C(=O)NCCCC(C)NC(=O)C=CCCC=C(C)C)C1 45464,N1(CC(=O)NC(C2(O)CCN(C(=O)CS(C)(=O)=O)CC2)C)C(=O)C(=O)N(C)C1=O 45465,Cn1nc2ccc(Br)cc2c1C1CCCN1C(c1cnc(C2CCCCC2)s1)=O 45466,c1(OC(C(=O)N(CC(C)NC(Cc2c(C)con2)=O)C)C)ccc(F)c(F)c1 45467,CS(=O)(=O)c1ccsc1C(=O)NC1CCC(CNC(C2(n3cncn3)CC2)=O)C1 45468,N1(C(CC(CCC)CC)=O)CC2(C1)CN(C(C1CC3CCC1O3)=O)CC2CO 45469,C(C(CC=C)C(=O)NCC1CN(C2CC2)C1)NC(Cn1ncc(C#C)c1)=O 45470,Cc1ccc(Cc2cn(C3CCCN(Cc4cc(C5CC5)on4)C3)nn2)cc1 45471,CC1(C)CCOC1CC(=O)NC1CCN(C(=O)C=C2CCCCC2)CC1 45472,C1(CC#C)(NC(=O)C(Cc2cnc[nH]2)NC(C2C3(CC3)C23CC3)=O)CCCCC1 45473,c1(C(=O)NCC2CC2NC(=O)C(O)CC2CCOCC2)cc(Cl)ccn1 45474,N1(C(CCCC)=O)CCC2C(CCCN2C(=O)CCC(C)(C)F)C1 45475,N1(CC(=O)NC(C)C)C(=O)C(c2ccccc2)N(C)C1=O 45476,c1(C(=O)NCC(C)(C)NC(=O)COC2CCCOC2)nncn1C1CC1 45477,C1(C(=O)OC)CCN(C(=O)CC(C(F)F)NC(=O)C2CC2)O1 45478,N1(C(C(CC)NC(C)=O)=O)CCC(F)(F)C(NCc2cc(Cl)ccc2Cl)C1 45479,C1(CNC(c2cc(C)sc2)=O)COC(C)(C)CN1C(=O)CCc1cncnc1 45480,C(=O)(N=c1ccn(C)[nH]1)c1ccc(-c2cccc(C(=O)NC)c2)c(C)n1 45481,CCC(CC)CC(F)C(=O)NC(CN(C)C)C(=O)NC1CCN(C2CC2)C1 45482,C(=O)(CS(=O)(=O)CCO)N(CCCNC(c1cn(CC(N)=O)nn1)=O)C(C)C 45483,C1(C(=O)NC(CN(C(c2ccoc2CC(=O)OC)=O)CC)C)C2CCCC12 45484,N1(C(C=C(C)C)=O)CCC(C2CC2)(CNC(=O)CC(C)P(C)(C)=O)C1 45485,C(CCCCC(=O)N1CCN(C(C2CCN(C)C2=O)=O)C(c2cn[nH]c2)C1)SC 45486,c1(C(N2CC(OC)CC(NC(COCCC)=O)C2)=O)csc2c1CCC(C)C2 45487,C1(N(C(c2ccc(CCC)s2)=O)CC)CCCN(C(C2(N(C)C)CCC2)=O)C1 45488,Cc1cc(CNC(c2sc(C)nc2C)=O)oc1C(=O)N(C)Cc1cscn1 45489,c1(CC(N2CC(N3CCN(C(C4C(C)OCC4)=O)CC3)C2)=O)ccc(F)c(F)c1 45490,c1(NC(c2cn(C(C)C)nc2)C)nc(N2C3CCC2COC3)nc2ncn(C)c12 45491,C1(C(=O)NCC(CNC(C(C)C(F)F)=O)CO)CCC(O)CN1C 45492,c1(C(N2C(C(N(C)CC3(O)CCCC3)=O)CCC(O)C2)=O)ccc2[nH]ccc2c1 45493,C(=O)(C1CCCc2nncn21)N1C(C(C)NC(C(C)OCCC(C)C)=O)CCC1 45494,CCCCS(=O)(=O)CC(=O)NCC(C)CNC(=O)COC(c1nccn1C)C 45495,c1(NCC23CC(C(=O)NC(=O)CCN4CCOCC4)(C2)C3)nc2ccccc2s1 45496,c1(C(=O)NC2CC(CNC(c3coc(O)n3)=O)C2)csc2ccc(F)cc12 45497,C1(CNC(=O)C=C(Br)Br)C2CC1N(C(C1C3CCC(F)C13)=O)C2 45498,C1(CC(=O)NCCN(C(Cc2n(C(C)C)cnn2)=O)C)CCCCN1C 45499,N1(C(C(=O)NCC)CCCCN(C)C)CC2CCC(C1)C2C#N 45500,N1(C(c2onc(C)c2C)=O)CCC2(CC1)CC2(C)C(=O)NCCOCCO 45501,C1(F)(C(=O)NCC(CC=C)NC(=O)C(C)COC)CC2(CCC2)C1 45502,c1(SC)ccc(CC(=O)NC2C3CCN(C(=O)C(N4CCC(O)CC4)C)C23)cc1 45503,c1(C(N2CC(CCNC(C3(C#C)CC(=O)C3)=O)(OC)C2)=O)cccc(N=[N+]=[N-])c1 45504,c1(-n2cc(C(C(C)C)CCN)nn2)c[nH]c2ccc(C(C)C)cc12 45505,C1(NC(CC2C(COC)C2(F)F)=O)CC(Cn2cc(CC(=O)OC)nn2)CC1O 45506,C(CO)(CCCCNC(=O)CC1CCCO1)NC(C1(OCC)CCOCC1)=O 45507,N1(C(C2C(C)OCC2)=O)C2CCC1CN(c1ccnc(C3CCCC3)n1)CC2 45508,c1(CC(=O)NCCC(=O)NC(COC)C2(C)CC2)ccc(CO)cc1 45509,N1(C(c2ccc(C)cc2F)=O)CCC2(CC1)CC2C(=O)N(C1CC2CCC1O2)C 45510,C12(C)CC(F)(F)CN1C2.c1(NC)ccc(C(=O)OCc2ccccn2)c(OC)c1 45511,Cc1[nH]c(=NC2CC(NC(c3cnc4ccsc4c3)=O)C2)ccc1C#N 45512,N1(C(c2c(CC)cccc2)=O)CC(N(C)C(C2C3CC(F)(F)CC23)=O)C2(CC2)C1 45513,c1(C(N2CCC(N(C(c3sccc3C)=O)CC)C2)=O)cnc(C)nc1C 45514,N1(CC(=O)N(CC(CNC(CCN(C(CC)CC)C)=O)O)C)OC(C)(C)CC1=O 45515,N1(C(c2cc(C)no2)=O)CCC2(CC1)CC2CNC(C1(C2CCC2)CCC1)=O 45516,CCCCCCCC(=O)NC1(c2nnnn2C2COC2)CCCC(C(F)(F)F)C1 45517,c1(CC)ccc(F)c(C(N2CCCC(C)(CNC(c3c[nH]c(=NC)s3)=O)C2)=O)c1 45518,C1(NC(C2(CC)CC2(F)F)=O)CCN(C(=O)CCNS(=O)(=O)CC)CC(C)(C)C1 45519,c1(C(=O)NC(CSC)(C)C(N2CCC3(CCO3)C2)=O)ccc(C)cc1F 45520,CC1C(NC(=O)Cn2cncn2)CCCN1C(=O)C(=O)Nc1cnn(C)c1 45521,C1(C(=O)Nc2ccccc2-n2cc(C3CC3)nn2)CCc2ccccc2C1 45522,N1(C(CCC(c2ccc(SC)cc2)=O)=O)CCS(=O)C(C)C1C 45523,N1(CCNC(C(CN(C)C)N(C)C)=O)CCC(NC(=O)C=CC(=O)N(C)C)CC1 45524,N1(C(Cc2cc(C)no2)=O)CCCC(C2CC2NC(c2cncc(C)n2)=O)C1 45525,C(=O)(C1=CCCCC1P(C)(C)=O)NCCCCN(C)C(C1Cc2nccn2C1)=O 45526,c1(C(C2CC2)NC(C(C)(C)c2ccccn2)=O)cccc(F)c1 45527,C1(CC(=O)NC(CC(=O)NC)(C)C)CN(C(=O)CC(C)(C)C)CC12CC2 45528,c1(C(=O)OC)ccc2[nH]nc(C(=O)NCCNC(=O)C(O)C(C)SC)c2c1 45529,C1(NC(C2N(C(C3(C)CC(C)OCC3)=O)C3C(C2)C3)=O)CC(C)N(C)CC1C 45530,C1(C(=O)NC2(OCc3ccccc3)CC2)CCCN1C(C1CCCC1)=O 45531,Cc1cc(C(=O)NCC(C)NC(=O)Cc2cc[nH]c(=N)c2)c(C)cn1 45532,C1(C)(CNC(c2c(C)coc2)=O)CN(Cc2ccc(F)cc2Cl)CCO1 45533,CC(CN(C(=O)CCn1cnnn1)C)C(=O)N(CC(=O)N(C)C)C 45534,N(C(=NCc1ccco1)NC1CN(C2CCOCC2)C1)Cc1nc(CC)on1 45535,C1(CC)CN(C(=O)Cn2cc(C)cn2)CCC1CNC(=O)CSC 45536,CC1C(NC(=O)C=Cc2cn(C)nn2)CCN1C(=O)CC1OCCO1 45537,Cc1ccc(NC(C2CN(C(=O)CNC=O)CC(C)(C)C2)=O)c(F)c1F 45538,c1(N2CCC(C)(CC)CC2)nc(N2CCC3C(CCN3C)C2)nc2sccc12 45539,C1(NC(=O)CC2NC(=O)NC2=O)CC12CCN(C(=O)C1=CCOCC1)C2 45540,C=Cc1cncc(C(=O)NCCC2CN(C(=O)C3=C(C)OCC3)CC(C)O2)c1 45541,C(=O)(C(C(=O)OC)OC)N1C(C(C(=O)NCCC=CC)(C)C)CCC1 45542,C1(CC(=O)NC(CC=C)C)CCCN(C(=O)C(C)(CO)OC)CC1 45543,c1(COC)cc(C(=O)NCC2C(Cc3cc(C(=O)NN(C)C)no3)C2(F)F)no1 45544,C=C(C)C1CN(C(=O)CC2CCCN(C(=O)Cc3cnns3)CC2)CCO1 45545,c1(NC(C23CC(C(=O)NC(CC=C)CO)(C2)C3)=O)cc(Br)ncc1[N+](=O)[O-] 45546,N1(C(CC(C)CF)=O)CCN(C(c2cccn2Cc2cccs2)=O)C(C)C1 45547,CCC(O)(CC(=O)NC1CCC1CNC(=O)Cc1ccon1)c1ccccc1 45548,C1(CC(N2CCC(NC(c3c(C)nn[nH]3)=O)C2(C)C)=O)COc2ccccc2O1 45549,c1(NC(C(C(C)OC)NC(c2csc(=N)[nH]2)=O)=O)cnn2c1CCCC2 45550,C#CCC(C)(C)C(=O)N1CCN(CC(C)NC(=O)C(C2CCOCC2)O)CC1 45551,C(CC(C)C)(C(=O)NCCC1(NC(C)=O)CN(C(=O)C(=O)NC(C)C)C1)OC 45552,c1(C(=O)NC2CC(CNC(CCOC(C)=O)=O)C2)ccn2nnnc2c1 45553,CN1CCC2C1CCCN2C(=O)C(C1CCN(C(c2n[nH]c3c2COC3)=O)C1)F 45554,C1(C(=O)NCC(CNC(C2=CC(C)(CC)C2)=O)(C)C)CC2CCC(C1)C2O 45555,CC1CN(C(=O)CC(C)c2ccccc2)CC1NC(=O)CC(F)(F)Cl 45556,c1(CNCC23C(CN(C(C4CC(O)C4)=O)C2)C3)cccc(F)c1Cl 45557,O=C(C1=C(Cl)CCCC1)NCC1(NC(C23CSCC2C3)=O)CCOCC1 45558,N1(C(CNC(c2c(C)occ2)=O)=O)CCN(C(=O)CC2(C3CC3)CC2)C(C)C1C 45559,C(=O)(C1=CCC(F)(F)CC1)N1CC(CNC(=O)C=CC2CCCO2)OCC1 45560,CP(C)(=O)CCC(=O)NC(c1cccnc1)C(=O)NCC#CC#CCO 45561,C1(N(C(=O)NC(C)C)Cc2onc(C)n2)C2CCC1CN(C(=O)CCC1CC1)C2 45562,C1(OC)CN(C(c2conc2C(C)(C)C)=O)CC1NC(=O)C=CSc1nc[nH]n1 45563,c1(C(N2CC(C)(NC(=O)Cc3cccnc3)C2)=O)cncc(N)c1 45564,N#CC1(C(=O)NCc2csc(C(N3CCC(C4CCCO4)C3)=O)c2)CCCC1 45565,C1(F)(CNC(C2C(CC)CCC2)=O)CCN(C(=O)Cc2ccc(Cl)cc2F)CC1 45566,C#CCC(C)(CC)C(=O)NCC(C)CNC(c1nccn1C(C)C)=O 45567,C1(CCNC(C(F)=CCC)=O)CN(C(=O)CCN2C(=O)CCC2=O)CC(C)O1 45568,c1(C(=O)Nc2n(CC)nnn2)ccc(Cl)c(C(=O)OC)c1 45569,N1(CCc2nc(C)sc2)CCCC(NC(=O)N(C)CC2COCCO2)C1 45570,N1(C(CP(C)(C)=O)=O)CCN(C(=O)CCCn2cccn2)CC1c1cn[nH]c1 45571,C(C)(CCC(=O)N1CCN(CCCCCNC(=O)COCCC(C)C)CC1)SC 45572,c1(CC(=O)NCCCC(C)NC(c2ccsc2)=O)cnccc1C(F)(F)F 45573,c1(C(N2C(CC)C(NC(=O)CC(=O)NC3CC3)CC2)=O)n[nH]c2c1COC2 45574,N1(C(c2cc(OCC)cc(F)c2)=O)CCC2(CCCN(C(=O)C(C)(C)CF)C2)C1 45575,c1(NC(=O)OC(C)(C)C)ccc2c(c1)CC(C)N2C(c1c(OC)cccc1)=O 45576,Cc1ccc2oc(C(=O)N(C3CN(C(c4cn(C)c(C(F)F)n4)=O)C3)C)cc2n1 45577,C12(C(N(CCSC)CC)=O)CCC(CC1NC(c1cc(OC)n[nH]1)=O)C2 45578,Cc1cc(C(N2CCN(C(=O)C=CC(=O)OC(C)(C)C)CC2C)=O)ccc1[N+](=O)[O-] 45579,CC(CCNC(C1(CNC(=O)CC2CCOC2=O)CCCC1)=O)C(C)(C)C 45580,Cc1cccc(Cl)c1S(=O)(=O)N1CCN(Cc2cc[nH]n2)C2CC12 45581,C1(C(=O)NC(CNC(C(C)SCC)=O)CC(C)C)COC2COCC12 45582,C1(C(N2C3CC(NC(c4n(CC)ccn4)=O)C(C3)C2)=O)CCc2nnc(O)n2C1 45583,C1(C(=O)NC2CC(NC(C(CCC)NC(C)=O)=O)C2)CC2CCCC(C1)C2 45584,n1(CCCOC)nc(CCCOC)nc1-c1ncccc1CSc1ccccc1 45585,N1(C(c2cnc(NC(C)=O)o2)=O)CC(NC(=O)C(C)(C)N2CCCCC2)C2CC12 45586,C1(C(N2CCOC(C(N)=O)C2)=O)CCOCCN1C(C1CC(=C2CCC2)C1)=O 45587,C1(Cc2nc(C(C)Sc3ccccc3)n(-c3ccccc3)n2)CCC(F)(F)CC1 45588,N1(C(CC(CC)C)=O)CC(NC(C2CC3CCC2CC3)=O)CC(C)(C)C1 45589,c1(-c2scc(C(=O)NCCCCC#C)n2)cnn2c1CCCC2 45590,N1(C(C2CC(N(C)CC)C2)=O)CC2CC(C(=O)NCc3snnc3C)C(C2)C1 45591,CCC(C(=O)NC1CCSC12CN(C(c1ccc(CC)nc1C)=O)C2)C(C)(F)F 45592,C12(C(N3CCC(N(CC#C)C(C4CCC(C)O4)=O)CC3)=O)CCC(N=[N+]=[N-])C1C2 45593,CCCC(C(O)C(=O)N1CC(OC)C(F)C1)NC(=O)CN1C(=O)CNC1=O 45594,CS(=O)(=O)c1ccsc1C(=O)NC1C2CC1N(C(C1(C#N)CC13CCC3)=O)C2 45595,C(=O)(C(O)C(C)(C)C)NCCn1cc(C(N(CC#C)C)=O)nn1 45596,C1(CN(C(=O)CN2CCOCC2=O)C)CCCN(C(C2CCCS2(=O)=O)=O)C1 45597,c1(CC(N2CC(OC)C(NC(C3CC(N(C)C)C3)=O)C2)=O)cc(Cl)ccc1Cl 45598,C(=O)(C1=COCCO1)N1CCC(CCCCCNC(C2CCCS2)=O)CC1 45599,c1(C(=O)NCC2N(C(C(C)(Cl)Cl)=O)CC2)cc(C2CC2)oc1C1CC1 45600,Cc1cccnc1C(=O)NC1CCCN(C(=O)C(O)c2ccsc2)C1 45601,C1(C(=O)NCCCNC(C(C)Oc2ccc(F)cc2)=O)CCc2ncccc2C1 45602,C1(C(=O)OCc2nnnn2-c2ccccc2)CCc2cc(F)ccc2O1 45603,CCCC(C(=O)N1CCCC1(C)c1cn(Cc2cnco2)nn1)OC 45604,N1(C(CSCCC(C)C)=O)CC(NC(=O)C(c2cnn(C)c2)O)C(C2CC2)C1 45605,CC(C)(C)C(C)(C)C(=O)NC1CCC(NC(c2[nH]nnc2C2CC2)=O)CC1 45606,C1(C(=O)NCC=CCNC(C(c2c(F)cccc2F)C)=O)CC2CCCC(C1)C2 45607,c1(C(=O)NC2(CC)CN(C(=O)Cc3ccccc3I)C2)nccc(OC)c1OC 45608,c1(CC)cncc(C(N2CC(CCNC(=O)C(CC)NC(N)=O)C(C)C2)=O)n1 45609,C1(C(=O)NC2CN(C(c3ccccc3Br)=O)CC2O)Cc2ccccc2CO1 45610,Cc1ccc(C=CC(N2CC=CC(C(=O)NCC3CCOC3C)C2)=O)cc1 45611,C(C1COC(C)(C)O1)=CC(=O)NC1CC(C)(NC(C(C=C=C)C)=O)C1 45612,c1(CC)cnc(Cl)nc1N(C)CCN(CCOC)C(C1CCC2CC2C1)=O 45613,CCCC(CCC)=CC(=O)NC1CN(C(=O)Cc2ncccc2C)C2CC12 45614,Cc1ccccc1NC(=O)CCC1(NC(=O)CC2CC(O)C2(C)C)CC1 45615,c1(C(N2CCC(C(F)F)(CNC(C3CCO3)=O)C2)=O)c[nH]nc1[N+](=O)[O-] 45616,N1(C(CNC(CCC)=O)=O)CCC(NC(C2CC2c2c(F)cccc2F)=O)C(C)C1 45617,c1(CC(N2CC(n3cc(CCSC)nn3)(C(=O)OC)C2)=O)ccc(O)c(F)c1 45618,Cc1ccc2nc(C(=O)NC3(CNC(c4nc(C)oc4C)=O)CC3)c(N)n2c1 45619,c1(NC(C)=O)ccccc1CCC(=O)NCCCN(C(=O)C(F)C1CCOC1)C 45620,C=C(C)CC(C(=O)NC(c1cncs1)C)NC(C1CC2CC(=O)C1O2)=O 45621,C(N=c1[nH]c(=NCC(C)(F)C(C)(C)F)[nH]c2cc[nH]c12)c1scc(COC)c1 45622,C12(C(=O)NCCC(O)C(F)F)CCC(CC1)N(C(C1(CO)CCCCC1)=O)C2 45623,C(C(C(=O)NCC(C)N(C)CC)NC(c1nc(Cl)cs1)=O)SCC 45624,c1(CC(=O)NC2C3CN(C(c4c(C)cc[nH]4)=O)C2C3)ccc2c(c1)CC(C)O2 45625,C1(C(=O)NC(CNC(c2cc(Cl)c(Cl)s2)=O)CO)CCC2CC2CC1 45626,c1(C(=O)NC(CC=C)CNC(=O)C(c2ccc(Cl)cc2)O)c[nH]c2nccc-2c1 45627,c1(OC(C)C)cnc(C(=O)NC2CCC(CNC(c3cc(N)ccn3)=O)C2)cn1 45628,C(=O)(C1=CCN(C(=O)C(c2cnn(C)c2)=O)CC1)NC(CC(CC)C)C 45629,CCCC(CC(=O)NC1CCC(OC)CC1)NC(c1cc(C#N)cn1C)=O 45630,c1(OCC(=O)NCCCN(C(=O)CCc2ccncc2)CC)cnn(C)c1 45631,C(=O)(CS(F)(F)(F)(F)F)NCC1(C)CCN(C(C(C)OC)=O)C1 45632,CN1CCC(NC(c2cocn2)=O)C12CCCN(C(C1NC(=O)OC1(C)C)=O)C2 45633,Cc1c(C(=O)NC(C)(C)CNC(=O)CC2(O)COC(C)(C)C2)cc(N)cc1O 45634,c1(OCCOC)ccc(C(=O)NCc2cccnc2NC(=O)C(O)CSC)cn1 45635,Cc1ccnc2ccc(CN3CCC(CCNC(=O)COc4ccsn4)C3)cc12 45636,c1(C(=O)NC2CC(C)(NC(=O)CCc3ccncc3)C2)ccc([N+](=O)[O-])cc1 45637,N1(C(c2ccc(C(C)C)cc2)=O)CCN(Cc2nc(=N)[nH][nH]2)CC1C 45638,C1(CC)CC2(CCN2C(c2cn(C)nc2Cl)C(=O)NC2CCCC2)C1 45639,C1(C(=O)NC(c2csnn2)C)CCN(C(=O)C(c2cnn(C)c2)=O)CC1(C)C 45640,N1(C(CC(C)O)=O)CC2CCC(N(C(=O)CCc3cnn(C)c3)C)C2C1 45641,CCC(C(=O)NC(CNC(c1cccc2c1CCO2)=O)CO)C(C)(F)F 45642,c1(CC(=O)NCC2C3CN(C(C4OCCN(C)C4)=O)C2C3)ccnc(Cl)c1F 45643,C1(C(=O)NC2(CNC(c3csc4nccn34)=O)CCCC2)CCCCC12CCC2 45644,CCCCCCC(C)NC(=O)C(=O)Nc1cc(-c2ccccc2)nn1CC 45645,N1(C(Cc2cc(C)on2)=O)CCC(CNC(c2c(CO)noc2C)=O)C(F)(F)C1 45646,Cc1c(C(=O)NC2CC2NC(C2(c3ccno3)CCC2)=O)sc2cccc(F)c12 45647,C=CCCCCC(=O)NCC#CCNC(=O)C(S(C)(=O)=O)C1CC1 45648,CS(=O)c1ccc(CC(N2CCC(NC(C3CC(C)(O)C3)=O)C2)=O)cc1 45649,c1(C(=O)NCC2CC(OC)CN2C(=O)C(O)CCSC)cc(S(N)(=O)=O)oc1C 45650,N1(C2CCN(C(C(C)(C)OC)=O)C2)CCN(C(=O)CC2(C(F)(F)F)SCCS2)CC1 45651,c1(CC(=O)NCC(C)(CO)NC(=O)CC2OCCC2(C)C)cccc(Cl)c1 45652,C1(C(=O)NCC2C=CC(NC(C(C)c3ccsc3)=O)C2)CC2(C1)CC2(F)F 45653,C1(C(=O)Nc2ncc(Br)cc2OC(F)(F)F)CCc2n[nH]cc2C1 45654,c1(SC)ccc(NC(c2nc(C(=O)Nc3cnc(C)nc3C)cs2)=O)c(F)c1 45655,Cc1nccnc1C(=O)N(C)CCNC(=O)CC(C)Cc1cccc(F)c1 45656,N1(C(c2ccc(COC)o2)=O)C2CCC1(CNC(C1CC(SC)C1)=O)CC2 45657,C12(CC(=O)NCCC3CCN(C(=O)CCc4ccncc4)C3)CCC(CC1)OC2 45658,Cc1c(C(N2CCCC(N(C(=O)C#CC3CC3)C)C2)=O)cc(N)cc1O 45659,C(CC1CCCO1)N=c1[nH]c2ccc(S(=O)(=O)N3CCCC(CO)C3)cc2[nH]1 45660,CC1(C)COC(C(=O)NCC2CCC(C(=O)NCCCN3CCCC3=O)CC2)C1 45661,C(=O)(C(C)(O)C1CC1)N(CC(C)NC(=O)Cc1n[nH]cc1Br)C 45662,N1(CCCc2ccc(C)cc2)C(=O)CN(CCc2ccc(F)cc2F)C1=O 45663,C1(F)(C(N(CC)Cc2cccs2)=O)CCN(C(=O)Cc2nccn2C)C1 45664,n1(C(C)C)ncc(Cl)c1C(=O)NCC1CCC(F)(CNC(C2(C(N)=O)CC2)=O)C1 45665,N1(C(C(C)(C)n2cc(Cl)cn2)=O)CC2C(C(=O)NCCC3(C)CC3(F)F)C2C1 45666,C1(CCCC)CN(C(C2CC=CCC2C(=O)OC)=O)CCN1C(=O)C(C)CC 45667,c1(CC(=O)N(C(CNC(CSC)=O)C)CC)cc(Br)ccc1Cl 45668,c1(C(N(CCCOCCNC(c2ccc(SC)o2)=O)C)=O)nc(C)ccc1F 45669,C(CC(=O)N=c1cc[nH]cc1O)C1N(Cc2c(OC)nccc2)CCC1 45670,C1(C(=O)OCC(c2ccccc2C(N)=O)=O)(COC)CC2(C1)OCCO2 45671,c1(C(N2CCC(C(C)(C)C)(CNC(CS(CC)=O)=O)C2)=O)cccc(F)c1O 45672,c1(C2CCCN(C(c3ncc(I)s3)C(=O)NC(C)(C)C)C2)ccc(F)c(F)c1 45673,n1(CC)cnc2c(NCCCC(C)NC(=O)COc3ccon3)nc(Cl)nc12 45674,CCCCS(=O)(=O)CC(=O)NC1CN(C(=O)COc2c(Cl)cccc2Cl)CC1C 45675,c1(CNC(NCC(=O)OCC)=N)ncc(-c2ccccc2F)n1C 45676,C1(CNC(C2(SC)CC2)=O)CCCCN(C(c2ccc(N)cc2Cl)=O)C1 45677,CN=c1[nH]cc(C(=O)N(C(C)C(N2CC3C(C(N)=O)C3C2)=O)C)o1 45678,c1(C(=O)NCC2CC(C)(C)CN2C(c2cnccn2)=O)cc2ccccc2[nH]1 45679,c1(SCC(N2CC3C(NC(Cc4c(CC)con4)=O)(C3)C2)=O)cc(F)ccc1F 45680,Cn1ccc(C(=O)NCC2CCN(C(C3(n4cc(Br)cn4)CC3)=O)C2)cc1=O 45681,C1(NC(CC=CCC)=O)CS(=O)(=O)CC1NC(=O)CS(=O)(=O)NC(C)(C)C 45682,c1(OC)cc(C(N2CC3CC(NC(C4CCOC4)=O)C3C2)=O)ccc1C 45683,Cc1ccc(C2(C(=O)NCC(O)CCNC(c3csc(Cl)c3)=O)CC2)c(F)c1 45684,N1(C(c2ccc(C)cc2C)=O)CCCC(F)(CNC(=O)C(O)C(C)(C)C)CC1 45685,C1(C(=O)NCc2cc(C)c(C)s2)N(C(C2CCCC(CF)C2)=O)CCCC1(C)C 45686,N1(C(C(CCNC(C(CC=C)NC(C)=O)=O)O)=O)CCC12CN(C)C2 45687,c1(CC)ccnc(C(=O)NC(CNC(C2CC23CC(OC)C3)=O)CC(C)C)c1 45688,C1(CNC(CCC=C)=O)(C(=O)OC(C)(C)C)CCN(C(=O)C(O)CC(=O)OC)CC1 45689,N1(C(CCC(=C)Br)=O)CC2CC(C1)CN(C(=O)CCC(CC)OC)C2 45690,CCCC(C)(C)C(=O)N1CC(=O)CC1C(=O)NC(Cc1cnc[nH]1)CO 45691,C1(CNC(C2CC(SC)C2)=O)CCCCCN1C(c1cc(N)ccc1C)=O 45692,c1(OCC)ccc(C(=O)NC2CCCCC2CNC(c2ccnnc2O)=O)nn1 45693,C12(C(=O)NC3C(CNC(C(OC)OC)=O)C3)CC3CC(F)(C1)CC(F)(C3)C2 45694,c1(CN(c2cc(C)c(Br)cn2)C2C(c3cccc(C)c3)C2)ccc2cncn2c1 45695,C(C)(CC(=O)NC(c1nocc1C(=O)N(C)Cc1ccn(C)n1)C)SC 45696,Cn1ncc([N+](=O)[O-])c1N1CC(CCNC(c2cc(-c3ccncc3)no2)=O)C1 45697,CC12CC(CCO1)N(C(C1(NC(c3ccc(C#N)s3)=O)CSC1)=O)C2 45698,n1(CC(=O)NCC(C)(C)NC(C2C(OCC)C2)=O)c(C)cc(O)cc1=O 45699,N1(c2nnc(C)s2)CCC2(CCN(C(c3ccn4ccnc4c3)=O)CC2)CC1 45700,C(=O)(CCCS(N)(=O)=O)N1CC(NC(C2(C#C)CCC2)=O)C(C)C1 45701,c1(-c2nc(-c3cc(C)oc3C)nn2C2CCOC2)ccc2nsnc2c1 45702,Cc1cnc(C(C)(C)NC(C2CS(=O)(=O)C2)=O)s1 45703,n1(CC)ccc(C(=O)N(CCCNC(c2cc(C)cs2)=O)CC2CCCC2)n1 45704,C1(N(C(c2cncc(C(=O)NC3(C(C)CCO)CC3)c2)=O)C)CCN(C)C(C)C1 45705,C(C(C)CC(F)(F)F)NC(C=CC(C)NC(C1CCCN1C)=O)=O 45706,Cc1ccc(F)cc1C(=O)NCC(O)CCNC(c1csc(C(F)F)n1)=O 45707,C#CCC(CC)NC(=O)CCNC(C1(CO)CCCC1)=O 45708,C1(NC(CN2C(=O)NCC2)=O)CCN(C(C2CC3C=CC2C3)=O)C12CCC2 45709,C1(CN(C(C(n2c(C)ccn2)C)=O)C)CN(C(=O)CC2CCCC2)CC12CC2 45710,c1(C(=O)NC2CCCN(c3ncc(C)cn3)C2C)cnc2c(C)cccc2c1 45711,S(=O)(=O)(c1cccnc1N1CCS(=O)CC1)NCC(c1ccc(F)cc1)CC 45712,N1(C(C=C(CC)CC)=O)CCN(C(c2cc(N)c(Cl)cn2)=O)C2(CC2)C1 45713,N1(C(c2coc(Br)n2)=O)CC(F)(F)CC1CNC(C1(F)CCOC1)=O 45714,C1(NC(c2cn(C)nn2)=O)CCN(C(=O)C(=Cc2cccc(F)c2)F)C12CC2 45715,C1(N(CCC)CC)CN(N2CC(OCC)C2)C1.OC 45716,C=C(Cl)CC(C(=O)N1CCC(n2ccnc2)C1)NC(=O)Cc1ccccc1O 45717,CCCCCCCCNC(=O)CC1CC(F)CN1C(c1cc(F)c[nH]1)=O 45718,c1(SC)cncc(C(=O)NCC=C2CCN(C(=O)CCn3cc(C)cn3)CC2)c1 45719,C#Cc1cc(OC)cc(C(=O)NC(C)(C)C(C)CCC)c1 45720,C1(NC(CCCOC(C)C)=O)CCC(CNC(c2csc(S)n2)=O)CC1 45721,c1(C(C(N2CCC(NC(C34CC(F)C3C4)=O)C2)=O)O)ccccc1Cl 45722,C1(C)(C(=O)NCCc2ccc(C)nc2)CN(C(c2ccsc2)=O)C(C)(C)C1 45723,N1(C(CCc2c(C)noc2)=O)CCC(NC(c2cccnc2)=O)C1C(C)(C)C 45724,C1(NC(C2CC3CCC2CC3)=O)CN(C(=O)C(C2CCCCC2)O)CC2(CC2)C1 45725,C1(C(=O)NC2C(NC(C3C(c4cn(C)nc4)C3)=O)CCC2)CCCCNC1=O 45726,Cc1ccccc1C1(C(=O)NC2COCC2NC(=O)CSC2CC2)CCOCC1 45727,C(=O)(C(CN(C)C)C(C)C)N1CC(F)(CNC(c2c(C)oc(CO)c2)=O)C1 45728,c12nn(C)c(Cl)c1C(=O)O2.Cc1cncc(CCNC(c2ccco2)=O)c1 45729,N1(C(COCc2ccc(NS(CCCOC)(=O)=O)cc2)=O)CC2CC1CC2CO 45730,C(C)(C)(C(F)(F)F)OCC(=O)N(CC(C)N(C(=O)Cn1cc(C2CC2)cn1)C)C 45731,N1(C(C=CC2C(C)C2(Cl)Cl)=O)CC2(CCN(C(c3cc(C(N)=O)no3)=O)C2)C1 45732,c1(OC)cc(NCC2CC(NC(C3CN(C)C(=O)N3)=O)C2)nc(OC)n1 45733,C=C1CCN(C(c2ccn(CCNC(=O)Cc3nocc3C)c2)=O)C1 45734,C12(NC(CN(S(CC)(=O)=O)C)=O)CN(C(C3CCCC(OC)C3)=O)C(CO)(C1)C2 45735,C1(NC(C2(C=C)CCC2)=O)CCN(C(c2c(C(F)(F)F)cnn2C)=O)CC1F 45736,Cc1c(CNC(=O)CCC2CCCN2C(=O)C(C)(O)C2CC2)nnn1C 45737,Cc1nn(C)cc1CC(=O)N(CCCOCCN(C)C(C1(C)CC=CCC1)=O)C 45738,N1(C(C)=O)CC(O)CC1C(=O)NC1CC(C)C(O)C1.c1(C(=O)N)ncccc1Cl 45739,C(=O)(C1=CCCCCC1)N1C(C)CC(CNC(=O)C(O)C2CCCC2)C1 45740,C1(NC(CCC(C)OCC)=O)CCN(C(=O)C(COC)COC)CC12CCC2 45741,C(=O)(C1=C(C)OCCS1)N1CCCC(C(=O)NC2(SC)CCC2)C1 45742,N1(C(C(=O)NCC(C)N(C(=O)C(N2CCC(C)C2)=O)C)C)CCOCC1 45743,C1(OC)CC(NC(=O)CCCCCc2ccccc2)CN(C(=O)CC(C)F)C1 45744,N1(C(C(CC)C(C)C)C(=O)NCCC2CC2)CCC2(CC1)C(C)(C)C21CCC1 45745,CC#CCCC(=O)NCC(C)(O)CNC(C1COCCN1CC(F)(F)F)=O 45746,N1(Cc2c(OC)cccc2F)CCc2sc(-c3cc(C)nn3C)nc2C1 45747,c1(OC)cc(C(F)(F)F)[nH]c(=NCC(C)NC(=O)C(F)C(F)(F)F)n1 45748,C12(C(N(C)CC3CCN(C(=O)C(O)CF)C3)=O)CCC(C(F)F)(CC1)CC2 45749,CON(CCO)C(=O)C(CCOCCO)NC(c1ccc(C)cc1O)=O 45750,N#Cc1ccc(N)c(C(=O)NCC2(F)CC(NC(=O)C(F)OC(F)(F)F)C2)c1 45751,C1(C(=O)OC)CC2CCC(C1)C2NC(C1OCCC1C)=O 45752,c1(C(N2C3CCC(NC(C=C(CCC)CCC)=O)(C3)C2)=O)cccc2ccnn12 45753,c1(C(=O)NCCC(C)N(C(c2[nH]cc(C)c2C)=O)C)onc2ccccc12 45754,c1(C(N2C(C(N3CCC(O)C3)=O)CC3CC32)=O)cccc(C(F)(F)F)c1F 45755,CC(C(=O)NCC1CN(C(=O)Cc2nnc(S)n2C)CCO1)S(N)(=O)=O 45756,C12(NC(C(C)Cc3ccc(Cl)cc3)=O)CCC(C1)N(C(=O)CCC1CCCC1)C2 45757,O=C(C#CC1CCC1)NCC1(CNC(c2ccc(C(F)F)o2)=O)CCC1 45758,Cc1cc(Cl)c(C(=O)NCC2(O)CN(C(=O)C(c3ccncc3C)C)C2)c(Cl)c1 45759,Cc1cn2c(CC(=O)NC(c3ccc(F)cc3)CNC(c3ccsn3)=O)csc2n1 45760,C(CC1=CCN(C(c2n[nH]c(C)c2N)=O)CC1)NC(C1(CC)CCOCC1)=O 45761,C1(NC(CC2CC(=C)C2)=O)CCN(C(C2CC3CC3CC2C)=O)CC1F 45762,C#Cc1cc(CNCCNC(=O)C(C)c2cccs2)cc(F)c1 45763,N1(C(C(C=C)O)=O)CC(NC(=O)CC2CCOC2)CC12CCOCC2 45764,C(=O)(CC(C)C(C)(C)NC(C1CC(=O)N(CC)C1)=O)N1CCC(C#C)C1 45765,N1(C(c2cn(C)nc2-c2ccncc2)=O)CC2CCCC1(CO)C2 45766,C1(NC(COC(CC)C)=O)CCOCC1 45767,c1(CC(C(=O)NCC(CSC)(C)C)NC(C23CC(CO2)C3)=O)ccccc1Br 45768,c1(OC)ccnc(NCc2c(C(=O)CN3CC(CO)OCC3C)cccc2)c1 45769,C1(CNC(C2CNC(=O)N2)=O)CCCN(C(C2CC3CC3C2)=O)C1 45770,Cc1nc(CNC(=O)C(C2CCN(C(c3cc(C4CC4)on3)=O)C2)F)c(C)[nH]1 45771,C(=O)(CCCC(C)(C)C)NC(CC#C)CC(=O)NC(CC1CC1)CC 45772,C1(CNC(c2cn(CC(C)C)nc2)=O)CC2CN(C(C3CC4CCC3O4)=O)CC12 45773,CC(CNC(=O)C(=O)NCC(F)F)(C1CCC1)NC(=O)NC1CCOC1 45774,C1(C(N2CCCC2C(=O)NCC2COCCO2)=O)(CC)CCCCC1 45775,O=C1CC2(CCN(C(C3CC(NC(=O)CCc4nc(O)n[nH]4)C3)=O)CC2)CN1 45776,C12(CNC(c3c(OC)nccc3)=O)CCCC1N(C(=O)C(C)NC(N)=O)CCC2 45777,N1(C(C2CC=CCC2)=O)CCN(C(C2(c3ccccc3)CC(F)(F)C2)=O)CC1 45778,c1(C(=O)NCC2CCN2C(=O)COc2ccsc2)ccncc1F 45779,C12(C(=O)NCC3OCCN(C(C4CN(CCC)C(=O)C4)=O)C3)CC(C1)S(=O)(=O)C2 45780,c1(C(N2CC2)=O)cn2cc(C)sc2n1.C(C(C)(C)CSC)NC(=O)CC1(CO)CC1.CO 45781,Cc1ccc(C(N2CC3CCC(C2)N3Cc2c(F)cncc2F)=O)c([N+](=O)[O-])c1 45782,c1(C(=O)NC2(CO)CN(C(c3ccnc(C)n3)=O)C2)cccc2nccn12 45783,C1(C(=O)NC(C2(CSC3CC3)CC2)C)CC(OC(C)(C)C)C1 45784,N1(C(CC=C=C)=O)CCC2C(CCCN2C(c2ccc3c(c2)CCOC3)=O)C1 45785,c1(CC(=O)OCC)ccc(CN2CCN(C(C#N)C(C)C)CC2)cc1 45786,C1(C(=O)NCC2CN(C(c3cc(OC)n(C)n3)=O)C2)CCCC(C)(C)O1 45787,Cc1nn2ncccc2c1C(=O)NCC1(CN(C(=O)CC(C)P(C)(C)=O)C)CC1 45788,CCC(CNC(=O)C(C)C)(CC)C(=O)NC1CC(C)N(C)CC1C 45789,Nc1nc(C(N2CC3CC(NC(c4cc(CCCO)on4)=O)C2C3)=O)ccc1O 45790,c1(C2(C(N3CC(CC(C)NC(c4nc(CC)oc4)=O)C3)=O)CC2)ccc(Cl)nc1 45791,C1(C(=O)NC(C2CC2(C)C)C)(CF)CCN(C(=O)C(C)C2CCOC2)C1 45792,Cc1c(C(N2CCCC2(C)CCC(=O)NC2(CC(C)(C)C)CC2)=O)ncn1C 45793,C(C(=O)N1CCC1C(=O)NCCc1ccnc(C)c1)(C(C)C)NC(C)=O 45794,Cc1ccc(CNC2CC2C(=O)Nc2ccc(C(N)=O)nc2)c(Cl)c1Cl 45795,C=C(Br)CCC(=O)NC1CCC(CNC(=O)C=C(C)C)C1 45796,C1(NC(=O)Nc2ccc(-c3[nH]c(=NC)sc3)cc2)CCC2CC2CC1 45797,C(=O)(C(=O)C(C)CC)N(C(CC)CNC(=O)C(C)CSC)C 45798,c1(C(=O)NCCC(=O)NCCNC2CC2c2cscn2)ccoc1C1CC1 45799,C1(O)(CN(C(=O)CC2CC23CC3)C)CCN(C(=O)Cc2cccc(Cl)c2)C1 45800,C(=O)(CCC(=O)NCC1CN(C(=O)CN2C(C)CCC2C)CC1C)NC 45801,N1(C(c2cc(C)sc2)=O)CC(NC(c2cc(C(N)=O)n(C)n2)=O)CC(C)C1 45802,CC1CN(C(c2ccc(CN(C)C)o2)=O)CC1CNC(c1ccsc1C#N)=O 45803,CC1CC(C(N2CCC(NC(c3ccc(C(F)F)cn3)=O)C(C)C2)=O)CC(C)O1 45804,S(=O)(=O)(CCC(=O)NC1CC(NC(=O)C(O)C(C)(C)C)C(O)C1)NC 45805,N1(C(COC(CC)C)=O)CCC1C(=O)NCCC1(CO)CC1 45806,c1(NC(C2CN(C)C2)=O)ccc(O)c(CO)c1.c12nc(c(C)o1)C(=O)NC2 45807,N1(C(c2c(SC)cccc2)=O)CC2CCN(C(=O)C(F)n3cccn3)CC2C1 45808,Cc1ccc2c(N3CCCC4(CC4)C3)nc(=NCC3CCC(C(N)=O)O3)[nH]c2c1 45809,c1(C(=O)NC2CCCC(NC(C3N(CC)CCC3)=O)C2)cc(C#N)oc1C 45810,CC1CCc2ncc(C(N3CC4CC(C3)N(C(c3occc3Cl)=O)C4)=O)n2C1 45811,N1(C(c2nc(N(C)C)oc2)=O)CCCC1(C)CNC(=O)CCS(C)=O 45812,C1(CNC(C(CC)C)=O)CCN(C(=O)Cc2cccc(NC(C)=O)c2)C1(C)C 45813,C12(C(=O)NCC(N(C(=O)C3=CCCSC3)C)C3CC3)CC(C)(C1)OC2(C)C 45814,C1(CNC(c2c(CC)n[nH]c2)=O)CC(C)(C)CCC1NC(=O)CN(C1CCC1)C 45815,C1(C(=O)NC(CC#C)C(N)=O)CN(C(C2CCC(=O)N(C)C2)=O)CCN1C 45816,Cc1ccc(CCC(N2CC3CC2(CNC(C2CC2C)=O)C3)=O)c(C)c1 45817,CC1CN(C(=O)CC2CN(C)C2)CCN1C(c1coc(C2CCC2)n1)=O 45818,Cc1ccc(CC(=O)NCCC2(O)CN(C(=O)C(C)N3CCCC3)C2)o1 45819,c1(C(N(CCCCN(C(C(c2ccnn2C)C)=O)C)C)=O)cc(O)nn1C 45820,C1(N(C(CSCC)=O)C)CCC2(CC1)CCN(C(=O)CC1CCCC(C)(C)O1)C2 45821,c1(C(N2CC(NC(=O)C=CCF)C2)=O)cc(F)cc2nc(S)[nH]c12 45822,c1(C(N2CC(NC(C3CCCN(C(=O)OC)C3)=O)C2)=O)ncc(Cl)cc1F 45823,N1(C(CC2CCN(C(CC(COC)(C)O)=O)C2)=O)CC2(COCC(=O)N2)C1 45824,c1(C(C)NC(=O)NC(c2c(Br)cn(CC)n2)C)cccc2cnccc12 45825,c1(OCCOC)ccc(-c2cc(F)ccc2S(=O)(=O)NCC2(Br)CC2(F)F)s1 45826,n1(C(C)C)cc(Br)c(COC(=O)C(C)NC(c2ccccc2)=O)n1 45827,c1(C2(CNC(C3(C)COC(=O)C3)=O)CC2)ccc(Cl)cc1F 45828,c1(C(N(C2CCN(C(c3ccco3)=O)CC2)CC#C)=O)csc2c1CCCC2 45829,c1(NC(C)=O)ccc(Cl)c(C(N2CCC(NC(C3(F)CCC3)=O)C(C)C2)=O)c1 45830,N1(C(C2N(C(C)=O)CCOC2)=O)CCCN(C(c2ccc(Cl)o2)=O)CC1C 45831,n1(CC)cc(-c2n[nH]cc2C(=O)NCC(C)N(C(=O)C(C)NS(C)(=O)=O)C)cn1 45832,C1(NC(c2c(CCC)occ2)=O)CN(C(c2ccnc(S)c2)=O)C2(CCOC2)C1 45833,CN1N=C(C(=O)N2CCN(C(=O)Cn3ncn(C)c3=O)CC2C(F)F)CCC1=O 45834,C1(NC(c2c(C)nc(CC(C)C)s2)=O)CC12CCC(NC(c1csnn1)=O)CC2 45835,C1(F)(C(N2CCC(NC(c3cc(OC)nn3C)=O)C2)=O)CC2(CCC2)C1 45836,C=C=C(C)CC(=O)N(C1CN(C(c2cc(-c3ccn(C)c3)[nH]n2)=O)CC1O)C 45837,N1(Cc2ccc(C)[nH]2)CCC(C(=O)Nc2cccc(Cl)c2O)C(O)C1 45838,N1(C(C(c2cn(C)nc2)=O)=O)CCc2ccccc2C1CCNC(C1(O)CC1)=O 45839,N1(C(CSCCOC)=O)CCC2CCN(C(=O)COCCN(C)C)CC2C1 45840,CCCCC(O)C(=O)NCCC1CCCN1C(c1csc(-c2coc(=N)[nH]2)n1)=O 45841,O=C(CS(=O)(=O)CCO)NC1CCC(CNC(c2ccc(F)cc2F)=O)C1 45842,n1(CC(=O)NCC(CC)NC(=O)Cc2ccn(C)n2)c(-c2cccs2)nnc1S 45843,C(=O)(C(C)C(F)(F)C(F)F)NC1CC(CNC(COCCOCC#C)=O)C1 45844,Cc1ccc(C(=O)NC(C(N2CC(C(N)=O)C3(CC3)C2)=O)c2ccoc2)cc1F 45845,C1(NC(C=CC(C)NC(=O)Cn2ccnc2)=O)CCCCC1(C)C 45846,CC1CCc2ccccc2N1CCC(=O)NCC(=O)N(C1CCCCCCC1)C 45847,C1(OC)(CNC(c2nocc2C)=O)CCN(C(C2COCCC2C)=O)C1 45848,N1(C(CC(N)=O)=O)CC2CC(NC(=O)CCN3CCC3)C1C2 45849,Cc1ccc(CN2CC(CC(=O)Nc3ccc(Br)cn3)C2)cc1[N+](=O)[O-] 45850,c1(OC)cccc(NC(=O)CC(C=O)NC2(C)CC(C)=NO2)c1 45851,C1(NC(CCCCCC#C)=O)CCN(C(=O)CC(C(F)(F)F)OC)C12CCCC2 45852,c1(CCC)ccc(CC(N2CC=CC(NC(c3cnc[nH]3)=O)C2)=O)cc1 45853,C1(CNC(C=C(C)C)=O)(NC(C2CNC(=O)N2)=O)CCC(F)(F)CC1 45854,c1(CC(=O)NCC2(COC)CCCN2C(=O)C=C2CCC2)ccc(Cl)nc1C 45855,CCC(CC)C(F)C(=O)NCC1CN(C(C2CC3(CCC3=O)C2)=O)C1 45856,c1(C(N(C(C)C(C)C)CC)=O)cc(C(F)F)cc(C)c1 45857,N1(C(c2c(OCC)nccc2)=O)CCCC(CO)(NC(=O)C(O)CF)C1 45858,N1(Cc2onc(SCC)n2)CCSCC1Cc1nccc(C)n1 45859,N1(C(C(C)=CC)=O)CCCC(C)(NC(C2CC2c2ccc(F)c(F)c2)=O)C1 45860,S(=O)(=O)(c1ccc(Br)cc1NCc1ccc(C)c(N)c1)NCc1c(C)nc(C)s1 45861,CCC(CC)(CCNC(=O)C=CC=C(Cl)Cl)NC(=O)CN1CCCCC1C 45862,C1(NC(C(=O)NCC(c2ccc(OC)cc2)O)=O)CCc2cn(C(C)C)nc2C1 45863,c1(-c2scc(OCC)c2)cccc2cc(C(N3CCCC4CCCCC34)=O)sc12 45864,C1(NC(c2cc(CC)n(C)n2)=O)CC2CC1N(C(=O)CCOC1CCOCC1)C2 45865,C(=O)(C(CCN(C)C)NC(=O)C=Cc1cncs1)NCC(C)(C)OCC 45866,C1(NC(c2c(C)nc(C(F)(F)F)o2)=O)CN(C(=O)C(O)C2CC2)C(C)(C)C1 45867,c1(C(=O)NCCN(CC(C)O)C(c2c(C#C)cn(C)n2)=O)cn2cc(C)sc2n1 45868,c1(C(=O)NCCN(C(C2CN(CCC)C(=O)C2)=O)C)cccc(F)c1O 45869,c1(NC)cc(C(=O)NC2CCN(C(c3cccc(F)n3)=O)CC2CO)cc(Cl)n1 45870,c1(N2C(Nc3ccc(NC(CNC)=O)cc3F)C(C)CC2)nc(Cl)nc2sccc12 45871,C1(NC(c2n(C)cc(N(c3ncc(C(F)(F)F)cn3)C)n2)=O)CCC(C2CC2)C1 45872,c1(C(=O)NC2(CCNC(C=COCC)=O)CCOCC2)ccc2n[nH]cc2c1 45873,c1(C(=O)NCC=CCNC(c2ccsc2Cl)=O)ccncc1O 45874,C(=O)(CCOC(C1CN(CC2CCC2)C1)=O)OC(C)(C)C 45875,N1(C(C23CCC(OC)C2C3)=O)CCN(C)CC1CNC(=O)Cc1nocc1C 45876,N1(C(C2CN(C)C2)=O)CCCC2CCN(C(c3cscc3Br)=O)CC12 45877,C1(CCN(C)C(C2C(Cl)(Cl)C23CC3)=O)CCN(C(C2(C3CC3)CCCO2)=O)CC1 45878,C1(OC)CN(C(=O)NC2CCCN(C)C2)CCC1F 45879,Cc1ccc(C#N)cc1NC(C1CCN(C(C2CCOC2(C)C)=O)CC1(C)C)=O 45880,C(=O)(CC(C)CC(F)(F)F)N(C(c1ccn(C(C)C)n1)C)C(C1CCCCC1)=O 45881,Cc1ccc(NC)c(C(N2CCNCC2)=O)c1.C(=O)(C(=O)N(C)C)O 45882,c1(C(c2n(CC=C)nnn2)NCC(CO)C(C)(C)C)ccc2c(c1)CCO2 45883,c1(CC(=O)NC2C(NC(CC(=C=C)C)=O)CCC2)c[nH]c2c(F)cccc12 45884,N1(C(CCCCC)=O)CCc2nc[nH]c2C12CCN(C(c1cccc(N)c1)=O)C2 45885,CC1(C)C2CCC1(C(=O)NCC1CC(F)(CNC(C3CC34CC4)=O)C1)CC2 45886,CC(C(=O)NCC1CCN1C(c1cccc(=O)o1)=O)C(F)F 45887,Cc1ccc2[nH]cc(CCNC(=O)NCC(N3CCC(CON)CC3)(C)C)c2c1 45888,C12CN(CCC1(F)c1ccccc1)C2.C1(c2nnc(CC)n2C)CC12CCOCC2 45889,c1(C(N2CCC(C(N(C3(CO)CCC3)CC)=O)C2)c2ccccc2)ccccc1 45890,Cc1cc(F)cnc1C(=O)NCc1c[nH]nc1C(=O)NCCCC(F)(F)F 45891,C1(NC(CC(C)F)=O)CCCCC1NC(c1cc(-c2ccco2)cs1)=O 45892,c1(CC(=O)OC(CCC=C)C)cc(Cl)cc2ccccc12 45893,c1(OCC(=O)NCC(F)CNC(=O)COOC2CCOC2)ccc(F)c(F)c1 45894,c1(CC)cc(C(=O)NCCC2CC(OC)CN2C(c2cnco2)=O)oc1CC 45895,Cc1ncsc1C(=O)N(C)Cc1cocn1 45896,c1(C(=O)NCCC2(NC(C3C(C)(C(F)F)C3)=O)CC2)ccnc(C2CC2)c1 45897,C(C(=O)NNC(=O)c1ccc(F)cc1)NC1(c2nnnn2C)C(CC=C)CCC1 45898,C(=O)(CCCCN(C)C(c1ccc(C)nc1)=O)NCc1scc(C)c1 45899,C(=O)(C#CC1CCCOC1)N1CC(C)N(C(c2coc3ccc(F)cc23)=O)CC1 45900,C1(O)(CCNC(=O)CSC2CCS(=O)(=O)C2)CCCN(C(C2(O)COC2)=O)C1 45901,c1(C(=O)NC2C(NC(=O)CSC3CCCCC3)C2)ccncc1.C1(=O)CN1 45902,N1(C(CCOC)=O)C2CCC1(CNC(=O)Cn1cc(C3(O)CCC3)nn1)CC2 45903,C1(C(=O)NCc2cc(C)nn2C)CCN(C(c2ccccn2)=O)CC1O 45904,N1(C(=O)CC2CCCCC2)CCCC(C2CN(C(c3cc(F)ccc3Cl)=O)C2)C1 45905,c1(CNC(C2(SC)CN(C(=O)CC3(C)OCCO3)C2)=O)cc(F)ccc1O 45906,N1(C(c2cccc(CC)n2)=O)CC(C2CN(C(C3(O)CC3(C)C)=O)C2)C1 45907,C1(C2CC2)(CNC(C(C)OCC#C)=O)CCN(C(=O)CCC(C)OC)C1 45908,C1(C(N2CC(CCC)C(C(N3CCCC3CC3CC3)=O)C2)=O)CC(=O)NC(=O)C1 45909,C12(C(N(CCNC(=O)C(c3ccc(Cl)cc3)(F)F)CC)=O)CCC(CC1)OC2 45910,C(=O)(C1CSc2ccccc21)NCc1c(OCC#C)nccc1 45911,N1(C(CC(c2ccc(F)cc2)NC(C2CCCCO2)=O)=O)CC2OCCOC2C1 45912,N1(C(C2(OC(C)=O)CC2)=O)CCC(C(N2CCOC(CN(C)C)C2)=O)C(C)C1 45913,C(C(C)(C)CNC(=O)CC1(C)CCOC1)N(C(COCC(=O)NC)=O)CC 45914,C=C(C)CCCC(=O)N1CCC(C(C)(C)NC(=O)C(CC)c2cccnc2)C1 45915,C12(C(=O)NCC(C)N(C)Cc3n(CC(C)C)ncn3)CC3CC(C(=O)N1)C2C3 45916,C=CCC(CNC(C1(CO)CCC1)=O)C(=O)N1CCOCC1CC 45917,Cc1cccc([N+](=O)[O-])c1NC1CC(CCNC(C2CC3(CSC3)C2)=O)C1 45918,C=CCC(CC)C(=O)N1CCN(C(=O)COc2cccc(F)c2F)CC1COC 45919,N1(C(c2c(O)ccc(C)c2)=O)CCC(C(=O)NC(C)Cc2cnc[nH]2)CC1(C)C 45920,C1(N(C(c2c(CC)ncs2)=O)C)CCN(C(C2(c3ccsc3)CC2)=O)CC1 45921,CCC(C(=O)NCCCNC(c1cccc(N2CCCC2=O)c1)=O)C(C)O 45922,C=C(Cl)CC(C(=O)NCc1cc(C)ccc1OC)NC(=O)CCC(C)OC 45923,c1(SC)cccc(O)c1CC1(CNC(C)(C)C)CC1.c12cc(cn1C)NC2=O.NC 45924,c1(CC)nc(N2CC(OCCN)C2)cc(Cl)n1 45925,Cc1ccc(C)c(CC(N2CCC(CNC(=O)C=C3CC3)C(C)C2)=O)c1 45926,C1(NC(CCOCC#C)=O)CCC2(CC1)CC(NC(c1ccccc1F)=O)C2 45927,c1(C(N(CCNC(c2c(CC)n(CC)nc2)=O)C(C)C)=O)cccc(C)c1F 45928,C1(=O)C(F)CC(C)(C)NC(=O)C2CC(C2)N1.C1(C(N)=O)(CN(C)C)CCCC1 45929,CC(CC(F)(F)F)C(=O)N1CCC(C)(CNC(=O)C(F)C(C)(F)F)C1 45930,CC1CC(CNC(=O)CC2(C)CC2(Cl)Cl)CN1C(c1n[nH]c(=N)s1)=O 45931,c1(CNC(C(C)(N(C(C(CC)n2ccnc2)=O)C)C2CC2)=O)cnc(C)n1CC 45932,N1(C(C2(CCC)CCC2)=O)CC2CCCC2(NC(=O)C=C(Cl)Cl)C1 45933,N1(C(N2CCCC(CC(=O)OCC)C2)=O)CCCNC(=O)C1CC 45934,C1(SC)CCN(C(=NCCCCl)NCC(=O)N(c2cnc(C)c(C(N)=O)c2)C)C1 45935,c1(C2(CC)CC2)ccc(C(=O)NCC(CO)NC(c2oncc2C)=O)cc1 45936,C1(NC(c2n(CC)ccc2)=O)CC2(C1)CC(NC(=O)CC13CC(C1)C3)C2 45937,N#Cc1c(Cl)nsc1NCC1CCN(C(c2cc(CN3CCCCC3)on2)=O)C1 45938,C=CC1(O)CCN(C(=O)C(CCOCC)NC(C2CCN(C)C2)=O)C1 45939,c1(C(=O)NC(c2n(CC)ccn2)C(=O)O)cc(C)cc(O)c1 45940,N1(C(C(C)NC(C)=O)=O)CCOC(CCNC(=O)CC2CC(C)C2)C1 45941,Cc1oc(C2CC2)nc1NS(=O)(=O)CC1CC1F 45942,C(C(=O)N(C(C)CC)C)(C(C)CC)NC(c1cc(CC)on1)=O 45943,c1(C(N2CCC(CNC(C3CC4(CC4)C3)=O)C23CC3)=O)cc2c([nH]1)CCCC2=O 45944,C#Cc1ccc(CNc2cccnc2C(=O)NC(c2ccccc2)CN(C)C)s1 45945,N1(C(c2cc(C)cc(O)c2)=O)CCC(C2(NC(C3(C(C)C)CC3)=O)CC2)CC1 45946,Cc1cncc(C(N2CCC(O)(C(C)NC(=O)CCc3ccncn3)C2)=O)c1 45947,C1(NC(C(N(C)C)C2CC2)=O)CCC(N(C)C(C2CC(=O)N(O)C2)=O)CC1 45948,c1(CNC(C(N(C(CN(CCC)C)=O)C)C2CC2)=O)cnc(C)cn1 45949,N1(C(=O)CO)CC2CCN(C(c3nn[nH]c3Cl)=O)CCC2C1 45950,c1(C(=O)NC(CNC(c2ccsc2)=O)C2CC2)cc2c(nn1)CCCC2 45951,c1(C(N2C(CNC(CC3C(C)=NNC3=O)=O)C=CC2)=O)cc(C)ccc1F 45952,c1(NC(=O)C(F)CC2CNC2)cnccc1CO 45953,C1(CNC(C(C)OCC#C)=O)CCCN1C(c1c[nH]nc1-c1cccnc1)=O 45954,N1(Cc2ncc(C(=O)NC(c3nc(C)oc3)C)cn2)CCC(CN(C)C)CC1 45955,c1(NCC2CCN(C(=O)C=Cc3ccccn3)C2)ncnc2c(Cl)cc(Cl)cc12 45956,N1C(=NCc2ccccn2)N2CCC(C2)NC1=O.c1(Nc2ccsc2)ncccn1 45957,CC#CCCCCN=c1nc(N2CCCC3(CCCC3)C2)c2c([nH]1)CCS2 45958,c1(CC)ccc([N+](=O)[O-])cc1C(N1CCC12CN(C(C1CCCNC1=O)=O)C2)=O 45959,C(=O)(C(C(C)(C)C)c1cc[nH]n1)N(CCCNC(C(C(C)O)N(C)C)=O)C 45960,N1(C(c2n(C(CC)CC)nc(C)c2)=O)CCCC(NC(c2coc(C)n2)=O)CC1 45961,C1(C(C)N(C)C(N2CCCCC2CON)=O)CCN(C)CC1 45962,C#CCC(C)(C(=O)NCC(C)(O)CO)NC(=O)CC(=O)NC1CC1 45963,C1(NC(c2occ(C)c2)=O)(CO)CCN(C(c2ccc(CC(C)(C)C)cc2)=O)C1 45964,N1(C(C2OCCN(C(C3(CC(C)C)CCC3)=O)CC2)=O)C2CCC1CN(C)CC2 45965,c1(C(=O)NCC(COC)C)cn2c(n1)CCN(c1ncnc3cc[nH]c13)CC2 45966,C(=O)(C#CC1CCOCC1)NCC(C(C)C)NC(C1CC(=O)N(C2CCC2)C1)=O 45967,c1(C(=O)NCC2C(NC(=O)Cc3cscn3)CC2)cc2ncccc2s1 45968,N1(C(C(C)NC(N)=O)=O)CC2(CC(NC(=O)C(C)(C)NS(C)(=O)=O)C2)C1 45969,CCCCC(CC)CC(=O)NC(C(C)N=c1[nH]ncs1)c1ccccc1 45970,C1(F)(CNC(C(C)n2cnnn2)=O)CCCN(C(C2(C)CCCC2(F)F)=O)C1 45971,c1(C(N2CCC(O)(CCNC(=O)C=CC3CCCCC3)C2)=O)cc(=O)cc(Cl)[nH]1 45972,c1(CC2N(c3n(CC(=C)C)c(C(=O)OC)nn3)CCCC2)c(O)cccc1Cl 45973,C(C(C)(C(=O)NC1CCCN(C(=O)C=Cc2nccs2)C1)OC)OC 45974,C(c1ccccc1)=CCC(N1CCC(CN(C(C(COCC)C)=O)C)C1)=O 45975,N1(Cc2onc(N)c2-c2nnc(OC)n2C)Cc2c(ccc(F)c2Br)C(C)(C)C1 45976,C(=O)(CCC(C(C)C)NC(c1c[nH]c(C)c1)=O)N1CCCC(OC)CC1 45977,N1(CC)CC(C(=O)N(C)Cc2ccccc2CNC(=O)C2=CCCC2)CC1=O 45978,Cn1ncc(C(=O)NC2CC3CC(NC(C4OCC4(C)C)=O)C2C3)c1S(N)(=O)=O 45979,C=CCC(F)(F)C(=O)NC1CN(C(=O)COCCOCCO)C2CC12 45980,c1(Cn2ncc(C(N3CCC(c4ncc(C)cn4)CC3)=O)c2)ccc(Cl)c(F)c1 45981,Cc1ccc(CC(=O)NC2CC(CNC(=O)Cn3ccc([N+](=O)[O-])n3)C2)c(C)c1 45982,CC1(C)CC(NC(=O)CC#N)CN1C(=O)CSCc1cccc(Cl)c1 45983,C1(C(N)=O)CCCC(NC(=O)C(=O)NCCOCc2ccccc2Cl)C1 45984,N1(C(COCC(=O)NC)=O)CCC(C(F)F)(CNC(C2CC(C)(F)C2)=O)C1 45985,CC1CC(CNC(=O)C(O)C2CCCC2)CN1c1nccc(C2CCCC2)n1 45986,N1(C(CC2CCC(NC(COCC(C)C)=O)CC2)=O)CCSCC(C)C1 45987,C1(C)(CCC(=O)N(CCC(C)(C)C)C)CCCN1C(=O)CCc1ncnn1C 45988,C1(CNC(C2(OC)CC(CF)C2)=O)CC(=O)N(C2CN(C(=O)C=C(C)C)C2)C1 45989,c1(CCNC(CCc2cc(C)on2)=O)c(C)n[nH]c1C 45990,N1(C(c2nccc(CC)c2)=O)CCN(C(C2CC(C)=NO2)=O)C(CC(=O)NC)C1 45991,N1(CCCCCCCOCCOCC)CCN(CC(=O)NCC=CCl)CC1 45992,Cc1ccc2nc(C)c(C(=O)N(C3CCN(C(C4CC(Cl)(Cl)C4)=O)C3)C)cc2c1 45993,C1(C(=O)NC2CN(C(c3c(O)ccc(CC)c3)=O)CC2O)CCc2cnnn2C1 45994,c1(N(C)C)ccc(C(=O)Nc2cccc(-c3nn(C)c(=O)n3C)c2)cc1[N+](=O)[O-] 45995,CCCCC(C)CCC(=O)N1CCC=C(C(=O)NCc2cnccc2Cl)C1 45996,C1(CNC(C(C=CCCC)O)=O)CC(C)CCN1C(c1ccc(NC(C)=O)s1)=O 45997,c1(C(CC(=O)OC)NC(c2c[nH]cc2C)=O)cccc2ccccc12 45998,C1(NC(c2c(=O)ccn(C)c2)=O)CCC2(CC1)CNC2 45999,N12CC3C(C3C1)N(C)CCC2=O.c1(C(C)C(=O)NC2CCCCC2)ccn(C)c1 46000,c1(CC(=O)OCC2C(OC)CC2)ccnc(O)c1.C(=O)C(O)CN1CCCC1 46001,C1(NC(c2c(OC)nsc2)=O)CCC12CN(C(=O)CCc1csc(=N)[nH]1)C2 46002,N1(Cc2cncc(NC(CN(C)C)=O)c2)CCN(C=O)CC1 46003,c1(CC(=O)NCC=CC(N2CCC(CF)CC2)=O)ccc2c(c1)CC2 46004,N1(C(C2(N(C)C)CCC2)=O)CCN(C(c2ccn3nccc3n2)=O)C2(CCC2)C1 46005,N1(C(C2(CCCC)CCC2)=O)CCC2(CCCN(C(=O)CNC(=O)OC)C2)C1 46006,C(=O)(C(C(C)C)OC)NCCC#C.N(CCSCC)(CCOC(C)=O)CC 46007,Cc1cc(C(=O)NCCOc2ccccc2C(C)C)c(F)cc1Cl 46008,C1(CC(C)NC(c2cc(F)n[nH]2)=O)CCN(C(C2(C)CC=CC2)=O)CC1 46009,N1(C(CC(=O)OC)=O)CCC2(CC1)CC(NC(=O)C(CC1CCCC1)C(C)C)C2 46010,Cc1ccc(F)c(CC(=O)NC2CCC(NC(=O)C(F)C3CCC3)C2)c1 46011,C1(C(=O)NCC(O)CNC(C2CCC(c3ccccc3)C2)=O)(CC)CCCC1 46012,N1(C(C)=O)CCC2(CCOCC2)C(NC(c2coc3c2C(=O)NCCC3)=O)C1 46013,c1(CN(C)C(C2CC(NS(C)(=O)=O)C2)=O)ccccc1CNC(=O)C(C)(C)OC 46014,C1(C(N2CC(CC(C)NC(C3=C(C)OCC3)=O)C2)=O)CCc2nc(O)[nH]c2C1 46015,CCCCCCCC(=O)N1CC2CCC(NC(=O)CCN(C)CC)(C2)C1 46016,c1(C(=O)NCC(CN(C(c2n[nH]c(C)c2C(F)(F)F)=O)C)O)ccnc(Cl)c1N 46017,CC1CCC(CN(C)C(C2(CNC(C3CCCC(CF)C3)=O)CCC2)=O)CC1 46018,C1(NC(C2CCCN(C)C2)=O)COC2(C1)CN(C(c1ncnc(O)c1Cl)=O)C2 46019,c1(C(N2CCC3CN(C(C4C(C=C)C4)=O)CC32)=O)cnc2ccccc2n1 46020,c1(OC)cc([N+](=O)[O-])ccc1CN=C(NCC(F)F)NC1CCCCC1C 46021,C(=O)(C1=CCC(NC(=O)CC2CCC2)C1)NCc1nccc(OC)n1 46022,CCC(Cc1ccccc1)C(=O)NCCN(C(=O)Cc1nncn1C(C)C)CC 46023,N1(C(C2(C)CC2(F)Cl)=O)C(CNC(C2CCCO2)=O)CC2COCC12 46024,c1(-c2cn(CC)c(=O)cc2)ccc2ccc(C(=O)Nc3ccc(Br)nc3)nc2c1 46025,CC#CC1CCN(C(=O)C=CC(C)NC(C2C3C4CCC(C4)C23)=O)CC1 46026,CC(CN=c1[nH]c(=NC(C)c2ncc[nH]2)[nH]c2ccc(Cl)cc12)N1CCCC1 46027,N1(C(C(C)N(C)C)=O)CC(CO)C2(C1)CN(C(C1CCn3ncnc3C1)=O)C2 46028,C(=O)(C(C)CC(F)(F)F)NCC1CC(OC)CN1C(c1c[nH]nc1C)=O 46029,C(=O)(CS(=O)(=O)CC(=O)OC)N1C(CNC(C(CC)=CC)=O)C(C2CC2)CC1 46030,c1(C(=O)NC(CCCCNC(C)=O)C)cnc2c(C)cnn2c1 46031,C1(C)COCCC1CN.c1(NC(=O)NC(C)(C)CC2CCOC2)coc(CO)c1 46032,C1(C(=O)N(CC(C)(O)C2CC2)C)(CC)CCN(C(=O)C(C)CC)CC1 46033,c1(C(=O)NCc2ccc(-c3nn[nH]n3)nc2)cccc2[nH]ncc12 46034,c1(-c2cn(C3CN(C(c4c(C)coc4)=O)C3)nn2)cccc(CO)n1 46035,N1(C(C2CCCOC2)=O)CC2(CCCCN2C(c2ccnn2CC2CCCC2)=O)C1 46036,c1(N2Cc3c(C)cccc3C2)[nH]c(=NCc2ccc(Br)o2)nc2scnc12 46037,C1(NC(c2nccc(C)n2)=O)CCC2CCN(C(=O)C=Cc3ccc(C)o3)C12 46038,c1(C(N2CC(C)c3c2cccc3)=O)ccc(S(=O)(=O)c2ccccc2)s1 46039,N(C(=NCCC(C)=O)NCC1SCCS1)CC1CCCN(C(C)=O)C1 46040,N1(C(C2(OC)CCSC2)=O)CC(CNC(=O)CCn2cncn2)C2(CCC2)C1 46041,c1(OCC(=O)NC(C(C)NC(C2CCCCC2)=O)C)cccc(Br)c1 46042,CC1(C)CC(CC(=O)NC(CO)C2CCC2)CN1C(=O)CC1CC(=O)C1 46043,c1(CCCC(=O)NCC2(NC(C3CCCO3)=O)CC2)ccc(Cl)c(Cl)c1 46044,c1(CC(C)C(N2CC3CN(C(C4(F)CC4)=O)CCC23)=O)cnc2ccccc2n1 46045,N1(C(C(c2nc(CC)cs2)OCC)=O)CCSC(CC)(CC)C1 46046,C1(CC(=O)NC(C2CC(NC(=O)C=Cc3nccs3)C2)C)CCN(C)C1=O 46047,C1(NC(c2ncn(C(C)(C)C)n2)=O)CCN(C(C2(C)CC2(Cl)Cl)=O)CC1(C)C 46048,c1(C(N2C(C)CN(C(=O)C(F)(F)CO)CC2)=O)cc2n(n1)CCCC2=O 46049,C1(C(=O)NCC2C(NC(=O)CCc3ccc(Cl)nc3)C2)CCOC(=O)CC1 46050,C1(c2n(CCOCC)nnn2)(NCC2(SC)CCC2)CCCC1C(C)C 46051,Cn1cnc2cc(C(=O)NC3C4CC3N(C(=O)C(C)(Cl)Cl)C4)ccc12 46052,C1(NC(C(C)N(C)C)=O)CN(C(=O)CC2CC2C)C2(CCOCC2)C1 46053,c1(OC)ccc2c(c1)C(Nc1ccc([N+](=O)[O-])cc1Br)CC2 46054,CN1CC(O)CCC1C(N1CC2(CNC(c3cnn[nH]3)=O)CC1CO2)=O 46055,C1(NCC(c2ccc(F)cc2)N2CCOCC2)CNC2(CCOC2)C1 46056,N1(C(COC(C)(C)C)=O)CC2CCN(C(C3CC=CC3)=O)C2C1 46057,C1(CNC(c2ccc(O)nc2)=O)CC2(CCN(C(C3(CF)CC3)=O)CC2)CO1 46058,Cn1cnc2sc(C(=O)NCC3(O)CN(C(C4(O)CCCCC4)=O)C3)cc12 46059,c1(C(N2CCC(NC(C(C)(C)F)=O)C2)=O)cc2ccc(Cl)cc2c(=O)o1 46060,N1(C(C(=O)NC2COC2)c2ncco2)CCOCC1c1cccc(F)c1 46061,C1(NC(c2ccccc2)COCC(C)C)CCCC(N)C1 46062,C1(CC=C)(NC(c2ncoc2C2CCC2)=O)CN(C(c2ccnn2C)=O)C1 46063,C(=O)(C1CCCc2n[nH]cc21)NCC(C)NC(C1CC(C)(c2ccccc2)C1)=O 46064,CC1CCN(C(=O)CCCc2ccncc2)CC1CNC(c1ccc[n+]([O-])c1)=O 46065,N1(C(c2c(C)csc2)=O)CC2CC(NC(=O)Cc3cc4ccccc4o3)C(C2)C1 46066,Cc1ccccc1N1CC(C(=O)N(CCCNC(=O)CC(C)F)CCO)CC1=O 46067,C=CCC(C(=O)NCCC(C)NC(c1cnn(C)c1CC(=O)OC)=O)C(C)(C)C 46068,CC1(C)CCN(C(c2ccc3sncc3c2)=O)CC1NC(=O)CCc1cncs1 46069,c1(C(C(=O)NCCNC(C(COC)COC)=O)C)ccc(S(C)(=O)=O)cc1 46070,CCC(=O)CCC(=O)N1CC(C)(CCC(N2CCC(N(C)C)(CC)C2)=O)C1 46071,CC(C)CC(O)CC(=O)NCNC1(O)CC2CCC1CC2 46072,O=C1C(=Cc2ccc(-c3ccc(F)cc3)cc2)Cc2ccc([N+](=O)[O-])cc21 46073,C(=O)(CCC(=O)NCC1CC(O)CN1C(c1cc(Cl)cn1CC)=O)NCC 46074,c1(C(=O)NCC2(NC(C3CC3F)=O)CCOC2)cc(Cl)cc(C(F)(F)F)n1 46075,c1(C(=O)NC(CC)(C)CNC(C2CS(=O)(=O)C2)=O)cc(F)c(F)cc1Br 46076,CC1(c2ccc(CNC(=O)CCc3cccc(C(=O)O)c3)cc2)NC(=O)NC1=O 46077,c1(C(=O)OC)ccccc1CCC(=O)NCC1(F)CN(C(=O)Cc2ccon2)C1 46078,c1(CNC2CC(NC(C(C(C)c3ccccc3F)O)=O)C2)cc(C#N)ccc1F 46079,C(CC(C(C)(C)C)NC(=O)Cn1ncn(C)c1=O)N(C(C(CC#C)C)=O)C 46080,C(CCC(C)(C)C(=O)NCC(C)CCCO)NC(c1c(C)ncnc1)=O 46081,CCCS(=O)(=O)C(C)C(=O)NC1CN(C(=O)CCCCCN(C)C)C2(CCC2)C1 46082,C1(NC(c2oc(C)c(Br)c2)=O)CN(C(=O)CCCCCNC(N)=O)C2(CCC2)C1 46083,N1(C(C2(C(=O)NC)CC2)=O)CCC2(CCCN(C(c3ccn(C)n3)=O)C2)C1 46084,c1(C(=O)NC2CC(CO)N(C(C3(C(N(C)C)=O)CC3)=O)C2)ccc2nn[nH]c2c1 46085,c1(C(=O)NCC2(O)CN(C(c3ccc(CC4CC4)s3)=O)C2)ccnc(Cl)c1Cl 46086,C1(CC(N2CCC(N(C(=O)Cc3cncc(C)c3)CC)C2)=O)CCCC2(CC2)C1 46087,N1(C(C(C(C)C)NC(C)=O)=O)CCC12CN(C(=O)C(C)NC(=O)C1CC1)C2 46088,C1(NC(c2cc3sccc3[nH]2)=O)CC2(NC(C3CC4(C3)CC4F)=O)COC1C2 46089,C12(C(=O)NCC(CC)O)CC(C)(CN1C(c1cc(COC)no1)=O)C2 46090,C(=O)(C1CCc2nccn21)N1C(c2ccccc2)CCN(C)CC1.c1(CN)cccs1 46091,C#Cc1ccc(C(=O)NC2CN(C(C3(C(=O)NC4CC4)CC3)=O)C2)cc1F 46092,C1(C(=O)NC2(c3ccn(C)n3)CC2)(NC(CC=CCC)=O)CCN(C)C1 46093,c1(OC)ccc(CN(C(=O)C(C)NC2C3CCOCC23)C)c(OC)c1 46094,N1(C(c2c(C(N)=O)nccc2)=O)CC2(CCN(C(c3csnc3Cl)=O)CC2)C1 46095,CC(C(=O)NO)NC(C1CC(C)N1C(=O)CCC1CCCCC1)=O 46096,N1(C(c2ncc(OC)nc2)=O)C2CCC1CN(C(C1CCC3(CCC3)C1)=O)C2 46097,C1(CNC(CCCCSC)=O)CCC2(CN(C(c3cccc(C)c3C#N)=O)C2)O1 46098,C1(C(N2CC(C)(CC=C)C2)=O)C=CCN(C(C23CSCC2C3)=O)C1 46099,C1(C(=O)NCC(C)(CO)NC(c2ccc(C)cc2)=O)CCCC2(CCC2)O1 46100,N1(C(=O)C=Cc2ccc(C(F)F)o2)CCOC2(C1)CN(C(C1CCOC1)=O)C2 46101,CC(=O)CCC(=O)N1CCC1(C)CC(=O)NC1CCC(C(N)=O)CC1 46102,c1(CNC(CCC2N(C(COCCSC)=O)CCC2)=O)cccc(O)n1 46103,C1(C(=O)NC(C(=O)NCCN(CCOC)C)CO)CC2(C1)CC2(F)F 46104,c1(OC(C)C)cccc2sc(NC(C3CC4CCCC4N3)=O)nc12 46105,C(CCCCC(=O)NC(C1(O)CCN(C(c2cc(CO)n(C)n2)=O)C1)C)OCC 46106,C(=O)(C(C)(C)C(O)C(C)C)N1CC2C(NS(CCOC)(=O)=O)C(CC2)C1 46107,C1(NC(C2C(C)(C)C2)=O)CCC2(CCN(C(c3ccc4cc[nH]c4n3)=O)C2)C1 46108,C1(C(N2CCN(C(CC(=O)NCC)=O)C(C(C)C)C2)=O)CC2OC(C)(C)OC2C1 46109,O=C1CC(C(=O)NC2CC3(C2)CC3C(N2CCn3nccc32)=O)=NN1 46110,C1(NC(C(C)(O)C2CCC2)=O)CCCN(C(=O)Cc2cccc(Br)c2)C1 46111,Cc1cc(CNCC2CCCCN2C(C2(O)CCSC2)=O)n(C)n1 46112,N1(C(C2(C)C(C)C2)=O)CCC(C2CC2)(CNC(c2ccc3[nH]ccc3n2)=O)C1 46113,C(=O)(C(F)CC(CC)CC)N1CCC(C(CC)NC(C23CCN(CC2)CC3)=O)CC1 46114,N1(C(C=CC=CC)=O)CCC2CC2(C(=O)NCc2n[nH]c3c2CCC3)CC1 46115,c1(OC)cc(Br)ccc1C(CO)NC(=O)NCc1oc(C)cc1C 46116,NC(=O)CC(C(=O)NCCC1CCCCC12CC2)NC(=O)CC1CCSC1 46117,c1(C(N2CC(CNC(C3C(OCC)C3)=O)(OC)C2)=O)c(O)nnc2c1COCC2 46118,c1(C2(CNC(c3ccsc3)CO)CCC2)ccccc1Cl 46119,C1(NC(C2CCC(=C)CC2)=O)C(C)CCN(C(c2ccc(Cl)c(F)c2F)=O)C1C 46120,C(=O)(C1=CCC(C)(C)CC1)N(C1CC2CN(C(C(CC=CC)CC)=O)C1C2)C 46121,c1(C(=O)NCC2C(C(=O)Nc3cnc(OC)nc3)C2)coc2c1COC2 46122,C(=O)(CCCC(F)(F)CO)NC1CC2CN(C(c3cncc(C#N)c3)=O)C1C2 46123,c1(OC(C)C)ccc(CC(=O)N(C2CCC(CNC(=O)CC(C)C)CC2)C)cc1 46124,c1(C(C(=O)NCCCSC)N(C2CCCO2)CC2CC2)ccc(-c2ccco2)cc1 46125,c1(CCOC)nc(=NC2CCCC(NC(C3(O)CCSCC3)=O)C2)s[nH]1 46126,Cc1cc([N+](=O)[O-])c(C)cc1C(N1CC2CN(C(=O)CN(C)C)CC12)=O 46127,C(C(CNC(=O)C(C)Cn1ccc(C)n1)S(C)(=O)=O)NC(C(COC)C)=O 46128,N1(C(c2c(C)[nH]cc2)=O)C(C(=O)N(C(C)C)Cc2ccco2)CCC1C 46129,O=C(C1CCCn2cnnc21)NC1CC(O)CN(C(C2C3(CC3)C23CC3)=O)C1 46130,c1(N2CCC(Br)=C(C)C2)nc(N(C)CCSC(F)F)nc2cc[nH]c12 46131,C1(NC(CNC(C(CC)C)=O)=O)CN(C(c2ccn(C)c2)=O)C2(CCCCC2)C1 46132,c1(C(=O)NCC#CCNC(CC2CCCC(C)C2)=O)c(F)cc(Cl)c(F)c1F 46133,Cc1ncc(C(=O)NCC2(NC(=O)C(C3CC3)N(C)C)CC2)cc1CC(C)C 46134,Cc1c(NC2CCN(CC(F)(F)F)C2)ncnc1N(C)CCOC1CC1 46135,c1(N2CCC(N(C)C(c3ccc(O)nn3)=O)C2)nnccc1C#N 46136,C1(C(N(C)Cc2ccc(CNC(C3C=C(C)CS3)=O)cc2)=O)CCCC(C)(C)O1 46137,c1(OC)ccc(C(N2CCCC2CC(C)O)C(=O)NCC2CCCO2)cc1Cl 46138,C(=O)(CC(C)(O)C(F)(F)F)NCC1N(C(c2ccc(CC)cc2C)=O)CC1 46139,c1(-n2c(-c3cnc(F)c(C)c3)nc(COCC)n2)c(C)cc(C)cc1C 46140,c1(C(=O)Nc2ccc(NCc3nccc(C)c3)nc2)ccc2nc[nH]c2c1 46141,c1(C(=O)NCC2CC(O)(CNC(C(OC)OC)=O)C2)nc(C)ccc1F 46142,C(=O)(C1CCCn2nccc21)NCC1C(NC(CN(CC(C)(C)C)C)=O)C1 46143,c1(NC(=O)NCCc2ccc(CC)s2)cnccc1C(F)(F)F 46144,c1(C(=O)NC2CCC(CNC(C(N3CCNC3=O)C)=O)C2)ccc(F)cc1N 46145,n1(CC(=O)N(C(CNC(Cn2cc(C(C)=O)nn2)=O)C)C)ncccc1=O 46146,C#Cc1cnn(C)c1C(N1CCC(F)(CNC(c2cncn2C2CC2)=O)C1)=O 46147,CC1CC(NC(C2CC(=O)NC(=O)C2)=O)CCN1C(=O)CCCn1cccc1 46148,c1(C(=O)NCC(CC)(CC)Nc2cncc(C#N)n2)ccc2nc[nH]c2n1 46149,c1(CC(C)C(=O)N2CCCC2CN(C)C(c2cc(F)c[nH]2)=O)ccc(F)cc1F 46150,C(=O)(CCC(C)NC)NC(CCN(CC)CC)C.N1(CCO)CCCC(C)C1 46151,C1(NC(CCC(=O)NCCC)=O)CCCN(C(c2ccccc2SC)=O)CC1F 46152,c1(C(CC)C(=O)N(C(C)CN(C(=O)COCC(=O)NC)C)C)c(C)noc1C 46153,C12(C(=O)OC(C)(C)C)CC3CC(CC(C3)C1)C2.CC1CC(C)OC1C(=O)NC 46154,C1(NC(c2c(COC)cco2)=O)C=CCN(C(c2cccc(N(C)C)n2)=O)C1 46155,c1(C(=O)NCCOCCN)ccc2c(c1)CCCC2.CN1C(=O)CSC1=CC=O 46156,C1(C(=O)NCc2ncco2)CCCCN(C(c2ccc(F)cn2)=O)C1 46157,N1(C(c2nc(C)oc2)=O)CCC(NC(=O)C(C2CCCN(C)C2)(C)C)C1C(C)C 46158,c1(C(=O)NC(C(=O)OC)C2CC(C(=O)O)C2)ccc2[nH]cc(C=O)c2c1 46159,c1(C(=O)NC2CCN(c3nnc(C(C)(C)C)o3)C2)cc2c(=O)[nH]ccn2n1 46160,O=C1COc2ccc(NC(=O)NC(c3cncs3)Cc3ccccc3)cc2N1 46161,C1(Cn2cc(CCC(C)O)nn2)(CNC(C2CCC(=O)NC2)=O)CC12CCC2 46162,CCCC(C(=O)N1CCN(C(C23CC(C)(CCO2)C3)=O)CC1CCO)C(C)C 46163,N1(C(c2cc(CC)c(CC)o2)=O)CC(C)CCC1CNC(=O)C(CC)(CC)OC 46164,c1(OCCC)ccc(-c2ccc(CC(N3CCOCC3)=O)cc2F)cc1C 46165,CC1(C)CN(C(=O)C=Cc2cscn2)C1C1CCNCC1.N1(CC2CCCC2)CCCC1 46166,C(=O)(CS(=O)(=O)CC1CCCN1)C(c1cn(CCS(CC)=O)nn1)(C)C.N 46167,N1(C(c2c(SCC)nccc2)=O)CC2(C1)OC1(CO)CC2(NC(=O)CCCF)C1 46168,CC(CCCNC(c1csc(F)c1)=O)NC(=O)C(c1ccccc1)F 46169,NC(C(=O)NCC1(F)CCCNC1)C1CCc2ccccc21 46170,C1(CC)CCCN(C(C23CCC(OC)C2C3)=O)C1C(=O)NC1CN(C)CCC1O 46171,C1(N(C)C)CCCCN(C(C23CC(CO2)N(C(=O)CCc2cn(C)cn2)C3)=O)C1 46172,Cc1cccc(C(C)N(C)Cc2cc[nH]c2)c1C 46173,C=CCCC(C(=O)NC(C1CCC1)C1CCC1)NC(=O)CC(C)OC 46174,c1(C(N2CCCC(O)(CNC(c3c[nH]c(=N)o3)=O)C2)=O)cc(=O)n2nccc2[nH]1 46175,C1(C(=O)NCCC(C)N(CCC)C)CC(C)CN1C(=O)CC1CCCC(=O)C1 46176,C1(CCNC(c2c(CC)c[nH]n2)=O)CCN(C(=O)C=C(C)C(C)(C)C)C(C)C1 46177,N1(C(c2ccc(CSC)o2)=O)CCC(C)C(N(C(=O)Cc2ncoc2C)C)C1 46178,CC1CCC(Cn2cc(C(C)NC(c3cnn(CCO)c3C3CC3)=O)nn2)CC1 46179,C(CC(C(=O)NC1CCCN(C(c2csc(C(F)F)n2)=O)C1)OC)OC 46180,CC1(C)OC(=O)NC1C(=O)NCC(c1cccc(Cl)c1)NC(=O)CCC(N)=O 46181,c1(OC)c(C(=O)NCC2(NC(C3CN(C4CCC4)C3)=O)CCC2)sc(Cl)c1Cl 46182,C=C(C)CC(C(=O)NCC12CC(CC)(CN1C(=O)C(CCC)OC)C2)NC(C)=O 46183,N1(C(c2ccc(C(C)C)s2)=O)CCC2(CC2NC(=O)C2=C(Cl)CCC2)C1 46184,N1(CCC(=O)N(C(C)CNC(C2(N(C)C)CCCCC2)=O)C)CCSC(C)(C)C1 46185,C1(C(=O)NCC(C)(C)Nc2nc(C3CCCC3)ns2)CCc2c[nH]nc2C1 46186,C(=O)(C(CCSC)NC(=O)CC1CC2CC2C1)N(CCCC)CCCC 46187,C1(C)(C(=O)NCCCc2cn(C)nc2)CCCN1C(=O)C(N)=O 46188,C=C(C)CC(C(=O)NC1CC2(CCCC2)C1)NC(C1CCC(C)(C)CC1)=O 46189,C1(C(=O)NCCCCNC(c2cnn(C(F)F)c2)=O)CCCC(C2CC2)O1 46190,C1(C(=O)NCC(CC=C)NC(=O)C(c2ccc(F)cc2)CO)CCS(=O)(=O)CC1 46191,C1(CC(=O)N(CC(=O)NCCSCCC=C)CC)CCC(=O)C1 46192,C1(C(=O)NC2CCC(NC(c3cn(C)nc3Cl)=O)CC2)COC2(CCC2)CO1 46193,c1(CC)ccc2c(Cl)c(C(=O)NC(CNC(C3(C#N)CC(C)C3)=O)CO)sc2c1 46194,CN1CCCC(CC(N2CCC(CO)(NC(=O)COCc3ccccc3)C2)=O)C1 46195,c1(C(=O)OCC(=O)N(c2cc(C(C)=O)c(O)cc2)C)cc(F)c(F)c(O)c1F 46196,c1(C2(C(=O)NCCNC(C3C=CCN3)=O)CC2)cccnc1 46197,N1(C(C(CC#C)O)=O)CCC2CCC(C1)N2C(c1ccc(Cl)cc1Cl)=O 46198,C1(CCCC)CN(C(C2(C)CCNC2=O)=O)CCN1C(c1nnn(CC)c1N)=O 46199,C(=O)(C(CC(C)C)NC(C1CC2(CSC2)C1)=O)N1CCC(SC)C1 46200,c1(CC(C)C)cc(O)nc(Nc2ccc(OC(=O)CCCC(=O)N(C)C)cc2)n1 46201,C1(NC(c2cc(Br)no2)=O)(CO)CN(C(c2ccnn2CC(F)F)=O)C1 46202,N1(C(c2c(CC)n(C)cc2)=O)CC(C)CN(C(c2cc(=O)cc(Cl)[nH]2)=O)CC1C 46203,CCCCCCCCC(C)CC(=O)N1CC(CO)(NC(=O)C=C(C)C)C1 46204,C1(CNC(C2(COC)CC2)=O)CC2CCC1N2C(=O)C(c1ccccc1OC)O 46205,N1(C(C2C(C)C2)=O)CC(NC(=O)CCc2cnccn2)C2(CCS(=O)(=O)CC2)C1 46206,N1(C(C2(COC)CC=CC2)=O)CC(CCNC(c2nn[nH]c2Cl)=O)OC(C)C1 46207,Cc1c(CNC(=O)NCc2cn(CCl)nn2)cccc1Br 46208,C=CCC(C)(CC)C(=O)N1C2CCC(C2)C1CC(=O)NCCn1cnccc1=O 46209,C1(OC)(CNC(C2(CO)CN(C(=O)CC(C)O)C2)=O)CCOC1 46210,C1(CC(=O)N(CC(N2CC(O)(CC=C)C2)=O)CC2CC2)CCC(=O)NC1 46211,c1(NC(C2(C)CN(Cc3cncnc3)C2)=O)ccc(F)c(F)c1Br 46212,C1(NC(=O)C(F)=C2CCC2)CCN(C(C2CC(O)(C(F)(F)F)C2)=O)CC1CO 46213,C1(NC(c2cc(CC)sn2)=O)CCCCC1CC(=O)NCCC(O)C1CCC1 46214,C1(CNC(C2CCOC2)=O)CCCCN1C(=O)CCC=Cc1ccccc1 46215,c1(C(N2CC(C(=O)NCC3C(OCC)CCC3)C2)=O)cc(CS(C)(=O)=O)c(C)s1 46216,N1(C(=O)CCCn2cccc2)CCN(C(=O)Cc2cc(F)cc(Cl)c2)CC(O)C1 46217,C12(CNC(C(CC)=CCCC)=O)CC(NC(=O)C(C)=CCC)(C1)C(C)O2 46218,c1(OCC)nc(N2CCN(CCN(C)C(C3CSCN3C)=O)CC2)ncc1Br 46219,N1(C(CCC2CCC(C)O2)=O)CCC2CC(CNC(c3cnoc3)=O)CCC2C1 46220,c1(C(=O)NCC(CC)NC(=O)C(c2cccc(C)c2)C)c2c(nn1C)CCSC2 46221,C1(C(N2CCC(C(C)C)(C(=O)NC(C)CC(C)(C)O)C2)=O)CCC2(CC1)CC2 46222,CCCCC(C)(F)C(=O)NC1CC1CNC(=O)C=Cc1ccc(Br)s1 46223,Cc1ccc(OC(C)C(N2CC(CNC(C3(C#N)CCCC3)=O)C(C)C2)=O)cc1 46224,c1(N2CCC(C(C)NC(C(c3cc(C)sc3)(F)F)=O)C2)ncnc2cnn(C)c12 46225,CC(C)CC(C)CC(=O)NCc1cc(C(=O)Nc2cncc(C(C)C)c2)ccn1 46226,c1(OC)ccccc1S(=O)(=O)N1CC=CC1C(=O)Nc1cc(C)c([N+](=O)[O-])cn1 46227,N1(c2ncnc(=N)[nH]2)CCc2c(NC(C3CCCC(C(N)=O)C3)=O)cccc2C1 46228,C1(C)(CNC(C(C=C=C)C)=O)CN(C(c2nc(O)nc(O)c2OC)=O)C(C)(C)C1 46229,CC(C)(C(=O)NCC1CC2CC2N1C(=O)CCP(C)(C)=O)S(C)(=O)=O 46230,CCCCCC(F)C(=O)NC(Cc1cnc[nH]1)C(=O)NC1CC(C)(C)OC1(C)C 46231,c1(C(N2CC(C)N(C(c3ccc(F)c(Cl)c3)=O)CC2)=O)cc[nH]c(=N)c1[N+](=O)[O-] 46232,Cc1ccc(C2CC2c2nc(-c3ccc(N)cc3)nn2-c2cnnn2C)cc1 46233,N1(C(C2CCOC2)=O)CCC(O)(CNCc2cnc(-c3ccccc3)s2)CC1 46234,C(=O)(CS(=O)C(F)(F)F)NCC(C)(C)NC(C12CCC(F)(CC1)C2)=O 46235,c1(CNC(c2nc(C)oc2)=O)nc(CNC(=O)CC(C)CF)cc(O)n1 46236,CCCC(C)C(=O)N1CC(C(C)(C)O)(CNC(C2CC2c2conc2CC)=O)C1 46237,N(C1COCc2ccccc21)C(=O)C(c1ccccc1)Sc1ccc(Cl)cc1 46238,C1(C(=O)NCCC(C)(C)NC(C2C(C(=O)OC)CCO2)=O)CCCCC1(F)F 46239,c1(OC)cc(CNC(c2nnn(Cc3ccncc3)c2C)=O)cc2c1OCO2 46240,N1(C(c2n(C)c(S)nc2)=O)CC2CCN(C(C3CCc4nnnn4C3)=O)CC2C1 46241,N1(C(CCCN(C(=O)OC)C)=O)CCC(NC(C2CCCC2C)=O)C2(CCC2)C1 46242,c1(NC(COC)C)cc(=NCC2CC(OC)C2)[nH]c(CSc2ccccc2)n1 46243,CC1CC(C2CN(C(=O)C(CC(F)F)NC(c3c[nH]c(=N)o3)=O)C2)=NO1 46244,N(C(=NCCSCc1ccccc1)N1CC(C)S(=O)(=O)C(C)C1)Cc1cc(C)ncc1 46245,CC1(C)C(CNC(=O)Cc2ccnc(F)c2F)CCN1C(C1CSC1)=O 46246,Cc1cc(=O)c(C(N2CC3CC2(CNC(C2(F)CCCC2)=O)C3)=O)c[nH]1 46247,Cn1nc(C(F)F)cc1C(=O)NC1CCCN(C(c2cc(F)cs2)=O)C1 46248,c1(C(=O)NCCOCC(C2CCCC2)O)csc2c(Cl)cccc12 46249,N1(C(C(C)(O)C2CCC2)=O)CCN(C(c2n[nH]cc2Br)=O)CC(O)C1 46250,c1(-n2cc(CCNC(c3c(OC)nc(C)cc3)=O)nn2)ccc2c[nH]nc2c1 46251,C1(NC(c2cc(C)ncc2)=O)CN(C(C2CC3COCC3C2)=O)CC12CC2 46252,N1(C(C(CC=C)C)=O)CC2(C(=O)NC3CN(C)NC3=O)CCC1CC2 46253,C(CCC1CC1)(C(=O)NC1CC1c1ccco1)NC(C(C)n1ccnn1)=O 46254,Cc1cc(C(=O)NCC2CCCC2C(=O)NC(c2ncc[nH]2)C)ccc1O 46255,Cc1nc(=N)n(C2CCN(c3ccncc3C(F)(F)F)CC2)[nH]1 46256,Cn1cc(C(C)(C)C(=O)NC2CN(C(=O)CC3(C(F)(F)F)CC3)C2)cn1 46257,c1(C(N2C(C3(O)CN(C(CC=CC=C)=O)C3)CCC2)=O)cnc(C)c(C)c1 46258,C(=O)(C1OC(=O)c2ccccc21)NCCN(C(=O)C=Cc1cnn(C)c1)C(C)C 46259,N1(C(C2C(C)C2)=O)CC23CCCCC2(C1)CN(C(C1(C#N)CCOC1)=O)C3 46260,C1(C(=O)NC(C(C)C)CNC(C2COC3(C)CC2C3)=O)CC2COCC(C1)C2 46261,c1(C(=O)NC2CCN(S(CCCC)(=O)=O)C2)cc(Br)c(O)c(Br)c1 46262,c1(Nc2c(C(=O)NCCC(=O)OCC)nccc2)cccc2cccc(C)c12 46263,N1(C(C(c2c(F)cccc2F)C)=O)CCCOC(CNC(=O)Cn2cccn2)C1 46264,N1(C(C2N(CC)CC2)=O)CC=CC1(C)C(=O)NOCC1CC1 46265,C(CCN=C(NCc1ccc2c[nH]nc2c1)NCC1CCCC(C(F)F)C1)SC 46266,c1(CC(=O)NC2(CC)CCN(C(c3cncn3C)=O)CC2)cnn2ccccc12 46267,C(=O)(C(C)(C)CS(C)(=O)=O)NC1C(C)CCN(C(c2ncnc3sccc23)=O)C1 46268,c1(NCCOCCN2CCN(C(C3C(OC)CCC3)=O)CC2)c(C)cccc1Cl 46269,N1(C(c2ccc(C(=O)OCC)o2)C(=O)NCC2CC2)CC2C(C1)C2(C)C 46270,C1(NC(c2n(C)c(S)nc2)=O)CN(C(c2c(F)cncc2Cl)=O)CC1(C)C 46271,n1(CC)nnc(C)c1COC(c1ncc(CC2CCN(C)CC2)s1)=O 46272,Cc1ccc(C(=O)NC23CC2CN(C(C2(C)CC=CC2)=O)C3)c(Cl)c1 46273,c1(CCN(C)C(=O)NCc2cnc(F)c(Cl)c2)ccc(C#N)cc1 46274,C1(NC(C(C)(Cl)Cl)=O)COC2(CCN(C(=O)COc3ccc(C#N)cc3)C2)C1 46275,c1(NC(N2CCC(N3CCNCC3)C2)=O)ccnc2ccc(Cl)cc12 46276,c1(C(=O)NCC2N(C(CNC(=O)OC)=O)CC(O)C2)cc(N)ccc1F 46277,C1(C(N2CCC(CN(C)C(c3cnc(N(C)C)s3)=O)C2)=O)CC12CCCCC2 46278,c1(NC(=O)NCC(CC(C)C)NC(=O)OCC)c(C)nn(CCO)c1C(F)F 46279,c1(C(=O)NC2CCN(C(C3(CCC)CC3)=O)CC2CO)n[nH]c2c1CCSC2 46280,C1(NC(c2cncc(C)n2)=O)(CNC(=O)C(F)C(C)C)CCC(F)(F)CC1 46281,C(=O)(CS(=O)C(F)(F)F)NCC(CCNC(C(CC)SC)=O)(C)C 46282,c1(CC)ccc(C(=O)N(C(C)CN(C)C(c2ccc(CN(C)C)o2)=O)C)c(C)c1 46283,C1(NC(C(C)N(CCC)C(c2cc(C(F)F)[nH]n2)=O)=O)CC2(CCOC2)C1 46284,Cc1noc2[nH]c(=N)c(C(=O)N(C3CCCOC3)C)cc12 46285,N1(C(C(C)C2CCCC2)=O)CC(O)(CN(C(=O)CCCN(C)C)C)C1 46286,N1(C(CCSCC)=O)CC2CCN(C(c3ccc(OC)c(N)c3)=O)CC2C1 46287,N1(C(C(=O)NCCCC)CC(C)CCC)CCC=C(c2ccco2)C1 46288,c1(C(=O)NCCCNC(C2CC3CCCC3C2)=O)cc([N+](=O)[O-])c(Cl)cc1Cl 46289,CC1CCCN(C(c2cc(C3CC3)on2)=O)C1CNC(c1cc(N)ccc1O)=O 46290,c1(OCC)ccc2[nH]cc(CN3C(=O)CCN(CCCCF)C3=O)c2c1 46291,c1(C(N2CC(NC(C(C)CC(C)(C)C)=O)C2)=O)cccc2c1C(=O)NC2 46292,N1(C(C2(CCCC)CCC2)=O)CC(C(=O)NCC(C)(O)CO)OC(C)C1 46293,c1(C(=O)NCC2C(NC(CCC(C)(C)OC)=O)CCCC2)cccc2ccnn12 46294,C1(NC(C(C)NC(c2ccccc2)=O)=O)CC2CN(C(c3coc(O)n3)=O)CC12 46295,CC1=C(C)CC(C)(C(=O)NCC2(CNC(C3CC(=O)N(C)C3)=O)CCC2)CC1 46296,CC1CCc2cc(C(=O)NCCN(C(=O)CC3(O)CCCCCC3)C)ccc2N1 46297,O=C(C1=CCN(C(c2cc(C3CC3)on2)=O)C1)NCC1CC1C1CCCC1 46298,c1(OCCOC)cc(CO)ccc1C(=O)NCC(C)(C)c1ccsc1 46299,N1(C(c2ccc(COC)o2)=O)CCN(C(C2CC(S(C)(=O)=O)C2)=O)CC1CO 46300,c1(NC(C)C)cnc(NC(=O)NOCCOCCO)cn1 46301,c1(CC)nc(C#N)cc(=NC(CCNC(=O)C(C)CC)C(C)C)[nH]1 46302,c1(CC)ccc(C(C)C(N2CCC(N(C(=O)CSCC(F)(F)F)C)C2)=O)cc1 46303,c1(C(=O)NCC2CCC(NC(C3(OC(C)=O)CC3)=O)C2)cnc2c(C)cccn12 46304,CC1(C)CCC(F)(F)CC1C(=O)NC1CN(C(c2cc[nH]c2)=O)CCC1CO 46305,C1(C(=O)Nc2scc(C(=O)OCC)n2)C2CC1N(C(c1cncnc1)=O)C2 46306,C(C(C)(C)CC(=O)NCC(O)C1(Cl)CC1)NC(c1c(C)n(C)cn1)=O 46307,N1(C(c2cc(SC)oc2C)=O)CCCC2(NC(c3cn[nH]c3)=O)CCCC12 46308,Cn1cc(CNC(C2(F)CCN(Cc3cc(O)ccc3O)C2)=O)c2ccccc12 46309,C(=O)(C(CC(C)(C)C)OC)NCCC1OCCN(C(CCNC(COC)=O)=O)C1 46310,c1(C(=O)NCC(CNC(c2c(OC)ccs2)=O)O)cccc(OC)c1OC(F)F 46311,C1(NC(c2[nH]cc(COC)c2)=O)CCN(C(c2nc(C)c(C)s2)=O)CC1C(C)C 46312,Cc1cc(C(N2CCC(CNC(=O)CSCc3ccccn3)C2)=O)nn1C(C)C 46313,c1(C(=O)NC2C(C)CCN(C(C(COC)C)=O)C2)cc2cccc(Cl)c2nc1C 46314,C1(C(=O)NCCCC(C)(C)NC(=O)CCSC2(C)CC2)Cc2cc(Br)cnc2C1 46315,C1(C(N(C2CCN(C(C3CC34CCOC4)=O)CC2)C)=O)CC(O)CN1C 46316,C1(CNC(=O)C=CBr)CCC(F)(CNC(=O)CCc2ncccn2)CC1 46317,N1(C(C2(C)CCNC2=O)=O)CCCC(NC(=O)CNC(c2ccccc2)=O)CC1 46318,C1(C(N2C(CNC(c3c(C)nc(CC(C)C)s3)=O)CC2)=O)Cc2cscc2C1 46319,c1(CC)nc(C)[nH]c1C(=O)NC1CN(C(c2ccn(C3CCCC3)n2)=O)C2CC12 46320,c1(C(N2CCC(CC(=O)Nc3c(C#N)nc[nH]3)CC2)=O)cnn2ccccc12 46321,CCCCC(CN=c1[nH]nc(C(F)F)o1)NC(=O)C1=CCCCC1 46322,c1(C(N(C2CCC(NC(COC(CC)C)=O)CC2)C)=O)cccc(Cl)c1O 46323,c1(C(CC)OC)ncoc1C.C1(=O)C(c2cscn2)NC(=O)CO1 46324,C(=O)(C1CCc2nccn21)N1C(C(=O)NCCn2c(C)ncc2)C(C)C1 46325,Cc1[nH]c2c(C(=O)NC3CC(NC(C4CCSC4)=O)C3)cccc2c1C 46326,C=C(C)CC(C(=O)NC1CCCN(C(C2CCCN2N=O)=O)C1C)NC(C)=O 46327,Cc1cccc(F)c1C(=O)NC1CCC(NC(C2(F)CC=CC2)=O)C1 46328,C(C(C(=O)NC(Cc1ccco1)CO)N(C)C)NC(C(C1CCC1)OC)=O 46329,Cc1cnc(C(=O)NC(C)(C)CNC(=O)CCc2cnc(C)nc2O)c(Br)c1 46330,c1(C(=O)NC2CCCCN(C(c3cccc(I)c3Cl)=O)C2)n[nH]c2ccccc12 46331,C1(NC(CCOCC#C)=O)CN(C(c2c(C)noc2CC)=O)CCC1CO 46332,N1(C(C(N2CCNC2=O)C)=O)CCC(C(=O)NCCN2CC3CC3C2)C1 46333,C1(CC(=O)NC(C2CCN(C(=O)C(C)C(C)C)CC2)(C)C)(COC)CCOCC1 46334,C1(NC(COc2ccc(OC)cc2)=O)CN(C(C23COCC2C3)=O)CC(F)(F)C1 46335,C(=O)(CC(CC(C)C)c1ccccc1)NC(CC)(C)CNC(=O)C1=CCCOC1 46336,C(=O)(CCCS(C)(=O)=O)NCC1N(C(c2cnc(C)nc2C(C)C)=O)CCCC1 46337,n1(CC)nc(C(C)C)cc1C(=O)OC.c12cc(n(C)n1)C(=O)NCCNC2=O 46338,C1(CN(C)C)CCCCN1C(C1CNCC1c1cncn1C)=O 46339,c1(C(=O)NCC(CO)NC(c2ncn(C(C)C)c2)=O)cn(C)nc1Br 46340,C(=O)(C1=NOC(c2ccc(F)cc2)C1)NC1(C)CN(C(c2ccoc2)=O)C1 46341,c1(C(N(C(CC)C(=O)OC)C)=O)coc2c1CN(C(=O)C(c1cncnc1)C)C2 46342,C(C(CC(C)C)NC1C(C)CCN1C(=O)COCC1CC1)NC(C=NC(C)=O)=O 46343,CC(C(CO)NC(C1CCO1)=O)NC(c1cc(Cl)ns1)=O 46344,c1(OC)cc(NC(=O)C(=O)NC(C)Cn2cnnc2)ccc1C(C)(C)C 46345,CCC(CC(=O)NC(c1cccnc1)C(=O)NCC(F)(F)C(N)=O)C1CC1 46346,C1(C(=O)NCC2CCN(C(=O)CC34COCC(C3)C4)C2)C2CCCCCC12 46347,C1(C(C)NC(=O)C=CC(=O)NC2CC2)CCCCN1C(C1CC2CC1C2)=O 46348,c1(C(=O)NC(C)C(C)(C)NC(c2ccn(CCO)c(=O)c2)=O)cc(O)cc(O)n1 46349,C(C)(c1ccco1)=CC(=O)N(C(C)C(=O)NC1CCC(C(N)=O)CC1)CC 46350,CCCCC(CC(=O)N(C(CSC)CC)C)NC(=O)C=C1CCC(C)CC1 46351,C(=O)(CC1COCc2ccccc21)NC(C1CN(c2cc(Cl)ncn2)CCO1)C 46352,C(=O)(CCCC(C)(C)C)N(c1ncccn1)CC.C12CCN(CC1)C(=O)CN2C 46353,O=C(C#CC1CCCO1)NC1CCN(C(=O)Cc2nsc3ccccc23)CC1F 46354,N1(C(C(C=C)O)=O)CCCOC(CCNC(=O)CCCn2ccccc2=O)C1 46355,C1(CNC(c2n(CC=C)ccn2)=O)CCCCN1C(c1cn(C)nc1C)=O 46356,CCC(CNC(C1CCOC(C)C1)=O)(CC)C(=O)N1CC2(C1)CC2(F)F 46357,N1(C(c2cccc(OC(C)=O)c2)C(=O)NCCCSC2CC2)CCOCC(C)C1 46358,C(=O)(C(F)CCC(C)(C)C)NCC1C(CC(N2CC3(CC(OC)C3)C2)=O)C1 46359,C1(CNC(C2N(CC)CC2)=O)CN(C(c2c(Cl)c(C)nn2C)=O)CCC1(F)F 46360,S(=O)(=O)(c1ccccn1)NC1CC(C(N2CCN(C(C)C)CC2C)=O)C1 46361,N1(C(C(CC(C)(C)C)F)=O)CC(CNC(C2(F)CCOC2)=O)CC12CCOCC2 46362,c1(CC)ncncc1C(=O)N(CCCNC(C1CCN1S(C)(=O)=O)=O)C(C)C 46363,C#Cc1ccccc1CN=C(NCC(F)F)NCC1(OCC)CCOC1 46364,N1(C(C2(CCOC)CC2)=O)CC=CC(NC(C23CCCC2(C(N)=O)C3)=O)C1 46365,C1(NC(Cc2cc(C)nn2C)=O)(CNC(C2COC(=O)N2)=O)CC2CCC1CC2 46366,CC(C)CCCC(=O)NCC1(C(N)=O)CN(C(C2CC(C)CCC2C(C)C)=O)C1 46367,c1(C(=O)NC(C)CCNC(c2cccnc2F)=O)c(F)cccc1[N+](=O)[O-] 46368,C(=O)(CCCS(C)(=O)=O)NC(CN(C(C1CN(C)CCN1C)=O)CC)C 46369,N1(C(c2sc(C)c(C)c2C)C(=O)NCCOC)CC2CCC(C1)C2O 46370,N1(C(c2cnc(C)o2)=O)CC(NC(=O)C(C)Cn2ccnc2)C2(CCCC2)C1 46371,NS(=O)(=O)c1ccc(C(=O)OCc2ccccc2C(=O)C(F)(F)F)cc1 46372,C1(C#N)(C(=O)NCCCN(C)C(c2cn(C)c(=O)n2C)=O)CC12CCCC2 46373,C1(C(=O)NCCCN(C(c2nccnc2N)=O)CC)C2CC3C(C2)C13 46374,N1(C(C(C)NC(C)=O)=O)CC2CCN(C(=O)CCN3CCOCC3)C2C1 46375,CCC(CC(=O)NC(C)CCN(C)C(c1cc(C2CC2)ccn1)=O)C(C)C 46376,C(N=c1[nH]nc(C(N)=O)s1)C1(NC(c2c(CC)occ2)=O)CCCCC1 46377,c1(CNC(C(C)OCC=C)=O)nc2c(s1)CCN(C(=O)C=CSc1nc[nH]n1)C2 46378,c1(C(=O)NCC2CCCN(C(C(C(=O)OCC)F)=O)C2)ccnc2nc(C)nn12 46379,CCCC(C)C(=O)N1CCC(N(C(=O)CCC#N)CC2CC2)C1 46380,CCCCCCC(=O)N1CCC(O)C(NC(c2cccc(N3CCCC3)n2)=O)C1 46381,C1(NC(c2ccc(N(C)C)nc2)=O)(CO)CCCN(C(=O)Cc2ccsc2Cl)C1 46382,c1(CC)ncc(C(=O)NCC(N2CCN(C(C3CNC(=O)N3)=O)CC2)C)c(O)n1 46383,C1(C(=O)NC2CCCN(C(COCCCOC)=O)CC2)Cc2ccccc2S1 46384,c1(C2(C(=O)NC3CCC(CCNC(CCC#C)=O)C3)CC2)cccc(F)c1C 46385,c1(CC)nc(=NCCOCCNC(c2ccn3nnnc3c2)=O)s[nH]1 46386,C(C)(C)(CN=c1[nH]c2cc(Br)ccc2o1)NC(Cc1c(C)noc1Cl)=O 46387,c1(CC(=O)NC2(CCCNC(C3C(C)(C)C3(C)C)=O)CC2)ccc(F)c(Cl)c1 46388,O=C(N=c1[nH]c2sc(-c3ccccn3)cc2s1)C1CC1NS(=O)(=O)CCl 46389,CC(CN1CCCC1S(=O)(=O)c1c(F)cccc1F)C(=O)NNC(=O)C(F)(F)F 46390,C#Cc1cnc(C(=O)NCC2C=CCN2C(c2cc3nc[nH]c3cn2)=O)c(C)c1 46391,S(=O)(=O)(c1ccc(Cl)s1)NC(C)C(N1CCC(N2CCCC2)CC1)=O 46392,N1(C(=O)C=CC(F)(F)F)CCOC(C2CN(C(=O)C=Cc3ccco3)C2)C1 46393,C1(C(=O)OCC(=O)C2CC2C2CCOC2)CSC2(c3ccccc3)CCC(=O)N12 46394,C(=O)(C1=CNC2=NCCC2=C1)N1CCN(C(C2C(OCC)C2)=O)CC1CC1CC1 46395,c1(N2CCCC(C)(CNC(c3n(CC)ccc3)=O)C2)ncnn2cccc12 46396,C1(CCCCC)CCC(C(=O)NC23CC(NC(c4cc(C(C)C)on4)=O)(C2)C3)O1 46397,C(c1ccc(Cl)s1)=CC(=O)NC(CNC(C1N(CC)CC1)=O)CCOC 46398,Cc1nn(C)c(C(F)F)c1C(=O)NCCNC(C12CCCC1CCC2)=O 46399,CCCS(=O)(=O)NC(C)C(=O)NC(C)CNC(=O)CN(C(C1CCCCC1)=O)CC 46400,C1(CNC(CCSC)=O)CCN(C(C2(C3CCCCO3)CCC2)=O)CC1C 46401,c1(C(C)C)ccc(F)c(NC(=O)NC(c2ccccc2Br)CF)c1 46402,N1(Cc2onc(CCOC)n2)CCCCC(NC(c2cccc(=O)n2C)=O)C1 46403,N1(C(CCCNC(=O)OC)=O)CC2(C1)CN(C(=O)CC1CC(C)(C)CO1)C2 46404,C1(NC(CCc2cnc(C)s2)=O)C=CCN(C(C2C(C)(C)C2(F)F)=O)C1 46405,c1(C(=O)NC(CN(C(CCOC)=O)C)(C)C)ccc2c(c1)CCC2(C)C 46406,N1(C(c2cnc(C)n2C)=O)CCC2(NC(=O)Cc3cncnc3)CCCC12 46407,N1(C(C(C)(Cl)Cl)=O)CCC(C)(CNC(c2cnn(CC3CCCC3)c2)=O)CC1 46408,N1(CC(=O)NC2CN(C(c3coc(Br)c3)=O)C2)C(=O)C2CC=CCC2C1=O 46409,C1(C(=O)NC(CC)(C)C2CC2)C2CC1N(C(=O)C(=Cc1cn[nH]c1)C)C2 46410,C1(COC)(CNC(c2cc(O)nn2C)=O)CCN(C(C2CC(O)CN2C)=O)C1 46411,c1(C(=O)NCC2CCCC(C#C)C2)coc2c1CN(C(=O)Cc1cncnc1)C2 46412,C1(CNC(c2c(CNC(=O)COCC3CC3)occ2)=O)CC12CCOC2 46413,C(=O)(C(C(=O)NC1(C)CC(NC(=O)C(=O)Nc2ccc(F)cc2)C1)OC)OCC 46414,C1(C(=O)NC(CC)CN(C(=O)CC2COC3CC2C3)CC)(OC)CCCCCCC1.CC 46415,C1(CCNC(=O)CC2CC3CC3C2)CN(C(C2(Br)CC2)=O)CCO1 46416,c1(CNC(N(C)Cc2nnc(-c3ccc(F)cc3)s2)=O)cc(S(N)(=O)=O)co1 46417,Cn1ccnc1CCC(N1CCC(n2cc(CNC(=O)CSC(F)F)nn2)C1)=O 46418,N1(C(CCc2ccc(C)o2)=O)CC(CNC(c2scc(C)c2Cl)=O)CC1C 46419,C1(CCNC(CC2CN(C)C2)=O)CCN(C(=O)C(N)=O)C1 46420,C1(NC(C(=O)NCC2(C(C(C)C)O)CC2)C)CCC=CCC1 46421,c1(C(CC)NC(=O)N)cccc(C#N)c1.N1(CCC(C)C(=O)OC)CC=CCC1 46422,c1(C(=O)NCC2CCN2C(c2cc[nH]c3nccc2-3)=O)cc(F)c(F)c(Cl)c1F 46423,c1(C(N(C2CN(C(C3CN(C(N)=O)C3)=O)CC23CC3)C)=O)n[nH]c2ccc(F)cc12 46424,C(N=c1[nH]c2cccc(F)c2s1)C1C(C)CN(C(c2cc3n(n2)CCCC3)=O)C1 46425,CCC(C)(C)CCCC(=O)NC1CN(C(=O)C(COC)N(C)C)CCC1(C)C 46426,CC1(CNC(c2ccc3ncc(Br)n3c2)=O)COCC2CCCN12 46427,C(c1ccc(OC(C)C)cc1)=CC(=O)NC(CN(C(CC(=O)NC)=O)C)CC 46428,C1(c2cn(Cc3cnn(CCCOC)c3)nn2)(C(=O)OC)CCOC1 46429,C12(C(=O)N)CCC(CN)(CC1)C2.C1(NC(C)=O)CC1.C(=O)NCCN(C)C 46430,N1(C(C(CCOCC)NC(=O)C=Cc2cnn(C)c2)=O)CC2CCN(C)C2C1 46431,c1(C(N2CCC(NCCO)CC2)=O)ccc(Cn2cc(C3CCOC3)nn2)cc1 46432,C(C)(C)(CC(C)NC(=O)CCN(C(c1ccc(C)s1)=O)CC1CC1)OC 46433,c1(C(N2C(C)CN(C(c3csc(C#N)c3)=O)C(C)C2)=O)ccc2c(c1)CCN2C 46434,C1(N(C(c2cncs2)=O)CC)CCCN(C(C2(C#N)CCOC2)=O)CC1 46435,N1(C(C(CC=C)OC)=O)CCC(CNC(c2cnc(COC)nc2O)=O)C(C)C1 46436,c1(CC(=O)NC2C(C)(C)CN(C(=O)C(F)F)CC2)ccc(O)c([N+](=O)[O-])c1 46437,C1(O)(C(=O)NCCCN(C(c2cc3ccncc3o2)=O)CC)CCCC(C)CC1 46438,N1(C(C2CC(=O)NCC2)=O)CC2(CCN2C(C2CC(F)(F)C2)=O)C1 46439,c1(C(CNC(CSC(c2cccc(C(F)(F)F)c2)C)=O)O)c(F)cccc1Cl 46440,CCC(CC)(CO)C(=O)NCC(C)(F)CNC(c1ccc(N)cc1F)=O 46441,Cc1cc(C(N2CCN(C(=O)Cc3cnsc3)C3CC23)=O)c(C)nc1C 46442,C#CCC(C)(C)C(=O)NC1CCCCC1NC(=O)Cc1ccsc1C 46443,c1(CC)nn(C)c(CC)c1CNC(c1ccc(F)cc1)c1nnnn1C1CCC1 46444,N(C(=NCC1CCC(=O)N1C)NC1CCC(O)CC1)C(COC)C 46445,C1(C(CNC(=O)C=CC2CCC2)C2CC2)CCN(C(C2C3CNC(=O)C23)=O)CC1 46446,Cc1cc(-n2cc(CNC(=O)CSCc3ccc(F)cc3Br)nn2)ccc1Br 46447,c12ccc(cc1)NC(=O)C(=O)O2.c1(SCC)ccccc1OCCCCC 46448,c1(C(=O)NCCCN(C(CSCC#C)=O)C)ncc(C)cn1 46449,C(CCCC(=O)N1CC(C(=O)NC(c2ccccn2)C)CCC1C)(OC)OC 46450,Cc1cc(C(=O)NCCOCCCNC(=O)CSc2nc[nH]n2)c(O)nn1 46451,C1(C(N(CC(C)(C)CNC(=O)CC2CCCC2(F)F)C)=O)CCN(C)S1(=O)=O 46452,C(=O)(CCC1=CCCCC1)NC1CC(C)(NC(C2N(C)CCC2)=O)C1 46453,C1(N(S(c2c(C)onc2)(=O)=O)C)CCc2ccccc2C1 46454,C(=O)(C1=NOC(CNC(c2cncc(O)c2)=O)C1)NC(C#C)C1CCC1 46455,CC(C)(CNC(=O)CC1CCCC(C2CC2)O1)CCNC(=O)Cc1ccns1 46456,N1(C(=O)NC2CC(COc3ccccc3)C2)CCCC2(CCCNC2=O)C1 46457,N(C(=NCCC12CCC(CC1)OC2)N(C)Cc1cnn(C)c1)CCC(=O)NC 46458,N1(C(c2cc(C)no2)=O)CC(C)(C)CC1CNC(c1nnc(C)cc1O)=O 46459,C1(Nc2cn(CC3C(=O)OCC3)nc2)CCN(C(C2CN3CCN2CC3)=O)CC1O 46460,c1(C(=O)NC2C(C)(C)CN(C(C3CCCOCC3)=O)C2)cnn2cccnc12 46461,Cc1cccc2[nH]cc(C(N3CCCC3C(=O)Nc3cccc(F)c3)=O)c12 46462,CC#CCCC(=O)NC1CC1NC(=O)C(C)CC1CCCCC1 46463,c1(NC(C2CSCCN2c2ccncn2)=O)cc(Br)cc2cn[nH]c12 46464,C12(NC(CC(C)NC(=O)C#CC3CC3)=O)CCC(CC1)C2(C)C 46465,C1(C(N(CCNC(=O)CC2CC=CC2)C2CC2)=O)CCOC(=O)N1 46466,C1(N(C(C(=O)N(C)C)=O)CC(=O)NC2CC(n3ccnc3)C2)CC(C#N)C1 46467,Cc1c[nH]nc1C(=O)NC(CO)C(=O)N1CCCC1 46468,C(=O)(CCC1CCc2ccccc21)N1CCN(C(c2c(C)scc2)=O)CC1CF 46469,N1(CC)N=C(C(=O)N2CCCC2C(C)(C)CNC(=O)CC2CC=CC2)CCC1=O 46470,C(=O)(C(CC1CCOCC1)NC(=O)C=CC1CCC1)NC(C(C)F)C 46471,Cc1cc(C(=O)NC(C2CCCN2C(=O)C=CC2CCOC2)C)c(Cl)cc1Cl 46472,c1(C(=O)NCCN(CCC)C(C2CCCCC2C(=O)OC)=O)cnn(C)c1CC 46473,CC(C)(C)S(=O)Cc1cccc(NC(=O)COC2CC2(F)F)c1 46474,N#Cc1ccc(C(=O)NCC2CCCC(CNC(=O)CNC(=O)CC(F)(F)F)C2)[nH]1 46475,c1(CNC(C=C(CC)CC)=O)cccc2c1CN(C(C1(COC)CCC1)=O)C2 46476,CCC1CN(C(C23CC4(F)CC(F)(C2)CC(C3)C4)=O)Cc2ccccc21 46477,CCC(CN(C)C)C(=O)N(CCCNC(c1sc(C)nc1CC(C)C)=O)CCO 46478,N1(c2nccc(Br)c2Br)CCC2CCCCC2C1 46479,CCC(C)CC(C(=O)Nc1cnc(C(C)C)nc1)NC(c1ccsn1)=O 46480,c1(C(=O)NCCNC(c2cnn[nH]2)=O)ccc(-c2ccccc2)cn1 46481,CC1CCCC(C(N2CCCCC2CNC(c2cc(=O)n(C)cn2)=O)=O)CC1 46482,C1(C(C)C)CC(CC(=O)NCCNC(c2c[nH]c(C(F)(F)F)c2)=O)CCO1 46483,c1(OCC#C)ccc(C(=O)NCC2CN(C(C3(O)CC(C)(C)C3)=O)CC2C)cc1 46484,CC1CCOC(c2ccccc2)CN1c1nnnn1CCCCCS(C)(=O)=O 46485,Cc1cc(C#N)cc(C)c1S(=O)(=O)NC(C)C1=CCNCC1 46486,c1(CNC(=O)CN2CCNC(=O)C2c2cccs2)ccc(F)cc1O 46487,c1(NC(=O)CC2CCCN2CC)ccc(N(C)CC2CCN2C(C)(C)C)c(C)c1 46488,Cc1ccc(Br)c(NC(c2cc(-c3cccc(N4CCOCC4)c3)cs2)=O)c1 46489,N1(C(C2CC2NCc2c[nH]nc2-c2ccccc2)=O)CCN2CCCCC2C1 46490,N1(C(c2cc(SC)oc2C)=O)CCC2(CCCN(C(=O)C=C3CC3)C2)C1 46491,Cc1nn(C)c(C)c1C(=O)NC1CN(C(C)C(=O)NCc2cccs2)CC1(C)C 46492,O=S(=O)(c1[nH]c(=NCc2csc(Br)c2)ccc1Br)NCC1CCC(F)(F)C1 46493,Cc1cc(C(=O)N(CCN(C)C(c2scnc2C2CCCC2)=O)C(C)C)no1 46494,C1(CN(C(=O)C(C2CC2)NC(C2(C(N)=O)CC2)=O)C)CC1(C)C 46495,c1(C(N2CCC(CNC(C(CC3CC3)OC)=O)C2(C)C)=O)cccc2ccnn12 46496,c1(-n2cc(CONC(C3ON=C(C)C3C)=O)nn2)ccc(F)cc1Cl 46497,N(C)(S(C)(=O)=NS(=O)(=O)c1[nH]cnc1Br)C(C#C)COC 46498,O=C(N=c1cc[nH]c(CCCO)c1)C1CCCN(Cc2cc(Br)ccc2I)C1 46499,C1(NC(N(CCC)CCC)=O)(Cc2ccc(F)cc2)CCNCC1 46500,N1(C(C(C(C)O)(C)C)=O)C2CCC1CN(C(c1cn(C3CC3)nn1)=O)CC2 46501,C1(C(N2CC(CC(C)NC(=O)C=CCN3CCOCC3)C2)=O)CCC2CC1CO2 46502,CC(C)(C(O)C(F)F)NC(C1CCCC1CNC(C1(n2cccc2)CC1)=O)=O 46503,Cc1cc(=O)oc(C)c1C(N1CC(NC(C2COCCN2CC2CCC2)=O)C1)=O 46504,CCCC(CCC)C(=O)NCc1cc(C)c(C(N2CCC2C2CCCOC2)=O)o1 46505,C#Cc1ccc(C(=O)NCC2(C)CCN(C(c3cncc(COC)c3)=O)C2)cc1 46506,c1(C(=O)NC2C(c3ccc(Br)cc3)(CC)C2)ccc(S(C)=O)c(F)c1 46507,C1(C(N2CCC(O)(CC)CC2)=O)CN(C(=O)Cc2cccc(F)c2)CCC1(C)C 46508,N1(CC(=O)NC(C(=O)N(CCOCC)CC)C2CCCO2)CCC(=O)CC1 46509,Cc1nc(C)n(Cc2cn(CCN(C(=O)CCC3CC(F)(F)C3)C3CC3)nn2)n1 46510,N1(C(c2ccn(COC)n2)=O)CC(OC)CC1CCNC(c1nocc1Cl)=O 46511,N1(C(c2c(C)ccnc2O)=O)CCCCC(NC(c2cn(C)nn2)=O)CC1 46512,C(=O)(CC1CCOc2ccccc21)NCC1C(NC(CCN(C)CCO)=O)CC1 46513,N1(C(C(c2ccc(F)cc2)C)=O)CC2CC1C2NC(=O)CS(C)(=O)=O 46514,CCC(CC(=O)N1CCC(CN=c2nc(C3CC3)[nH]s2)(C)C1)C(F)F 46515,C1(C(=O)OC)(OC)CCN(C(=O)Cn2c(C)c(C)sc2=O)CC1OC 46516,Cc1c(C(C(C)C)NC(N2CCOC(c3ccccc3)C2)=O)oc2ccccc12 46517,c1(CN(C(C(=O)NC2CCCCC2)C2CCSC2)C)ccc(-c2ccccc2)o1 46518,N(C1CC2(CN(C(c3ccnn3C)=O)C2)n2ccnc21)C(CC(=O)NCC#C)=O 46519,C(=O)(CC(O)C(C)C)NC1CCC(CC(=O)NCc2cc(C)ncn2)CC1 46520,c1(SCC(N2CC(CN(C(C3C(CC)OCC3)=O)C)C2)=O)ccc([N+](=O)[O-])cc1 46521,Nc1ccnc(C(N2CCC(F)(CNC(=O)CC3CSCCS3)C2)=O)c1Cl 46522,CCCCC(C(=O)NOC(C)CC)NC(c1nonc1N)=O 46523,c1(C(N2CCC(CN(c3nnc(C(C)C)o3)C)C2)=O)c(Cl)cccc1Cl 46524,N1(C(c2c(C)cccc2)=O)C(C(N)=O)CCCC1C 46525,C(=O)(C1CCCc2scnc21)N1C(C)CN(C(=O)COC2CCCCC2)CC1 46526,c1(C(=O)OCC)nccc(N(CCCNC(=O)Cc2cccc(F)c2)CC)n1 46527,c1(C(=O)NC2C(C=C)CN(C(=O)C(COC)OC)C2)cc(S(N)(=O)=O)c(C)s1 46528,c1(C(=O)NCC2N(C(C(F)OC)=O)CCC2C)cc(O)nc(C2CC2)n1 46529,N1(C(C=C(C)CNC(C2CCC(C)(C)C2)=O)=O)CC=C(CO)CC1 46530,CCC(C)CCCCC(=O)NCC(CC1CC1)C(=O)N1CC(C)C(F)C1 46531,C(CC(C)C(C)C)NC(C(CN(C)C)NC(Cc1scc(C)c1)=O)=O 46532,c1(C(N2CC(NC(c3c(C)ccs3)=O)C(C3CC3)C2)=O)cc2nc(Cl)ccc2o1 46533,N1(C(C2C(=C)C2)=O)CCn2c(CNC(C3C(Cl)(Cl)C34CC4)=O)nnc2C1 46534,C1(CNC(c2c(C)con2)=O)CCN(C(C2CCOC2)=O)CC1C1CC1 46535,N1(C(C(C)N(C)C)=O)CCCN(C(c2cc(C(F)(F)F)ns2)=O)CC1C 46536,c1(CN2CC3(CCC(C(=O)Nc4ccnnc4)O3)C2)ccc2nc(O)[nH]c2c1 46537,CCP(=O)(CC)c1ccccc1C(N1CCCC1CCNC(=O)CCC(N)=O)=O 46538,Cc1oc(C(C)C)cc1C(=O)NCCC(C(C)C)NC(=O)C(C)n1ccnn1 46539,Cc1ncnc(C(=O)NCC2CCC(NC(c3c(C)nn(C)c3Cl)=O)C2)c1C 46540,Cc1oc2ncnc(O)c2c1C(=O)NC1CCN(C(c2cc(Cl)no2)=O)CC1O 46541,n1(CCN(C)C(C2(C(F)(F)F)CCO2)=O)cc(C2CCCCO2)nn1 46542,c1(OC)cc(NC(=O)NCC2(O)CCOCC2)ccc1F 46543,n1(CC(=O)N(C2(CC(=O)O)CC2)C)cc(CC2CCCC2)nn1 46544,c1(CC)nc(N2CCCC(NC(=O)C(C)Cc3c(C)n[nH]c3C)C2)cc(Cl)n1 46545,N1(C2CCN(C(=O)CC3COCCO3)CC2)CCN(C(c2cnns2)=O)CC1=O 46546,C1(NC(c2cc(C(=O)OC)oc2C)=O)CC2CC(C1)N(C(c1n[nH]c(O)n1)=O)C2 46547,C1(NC(c2c(C)noc2N)=O)CN(C(c2ccccc2)=O)C2(CCOC2)C1 46548,CC(C)CCCC(C)C(=O)NC1CCC(C)N(CC(=O)NC(C)C)C1 46549,N1(C(=O)CCCn2cncn2)CC2CC2(C(=O)NC2CC23CCC3)C1 46550,C1(C(=O)OC)(C(C)C)CCCN1C(=O)CCN(C1CCCCC1)C 46551,CCC(C)C(C)CNC(C1CC(=O)CN1C(=O)CC1CCC(C)CO1)=O 46552,c1(C(N2CCC(c3ccc(Cl)cc3Cl)C2)C(=O)NC(C)(C)C)cc(O)cc(Cl)c1 46553,c1(C(=O)NC2C(CNC(CNC(C(C)C)=O)=O)COC2)cnn2cccc(Cl)c12 46554,c1(C(=O)OCC(=O)Nc2c(C)cccn2)cccc2c1C(=O)OC2(C)C 46555,N1(C(C=CC=CCC)=O)CCC2CCC12CNC(c1cn(CC)nc1C1CC1)=O 46556,c1(C(=O)NCC2COCC2NC(C=COCC)=O)cccnc1Sc1cccs1 46557,N1(c2nccc(SC)n2)C2CCC1CN(C(=O)C(C)Cn1ccc(C)n1)CC2 46558,n1(CC)c(=O)nc(O)c2c(C(=O)OCCCCCC(F)F)cc(C3CC3)nc12 46559,C12(C(=O)NC(CCNC(C(C=C=C)C)=O)C)CC3CC1C2C3(F)F 46560,c1(C(N2C(C)C(NC(=O)C(O)Cc3cnc[nH]3)CC2)=O)ccc([N+](=O)[O-])c(O)c1 46561,C1(CC(=O)NCc2ccc(C#N)s2)C2CCCC2N1C(c1ncccc1O)=O 46562,c1(C(=O)OC)ccc(C(=O)NCCCC(C)(C)NC(C2CCS(=O)(=O)C2)=O)cc1 46563,C1(NC(C(C2CCCC2)OC)=O)CC(O)(CNC(=O)CC2CCCN2C(C)=O)C1 46564,C(=O)(C1=CC2CCCC12)N1CCC(CNC(c2occ(C)c2)=O)(CO)CC1 46565,C(C(C(C)C)NC(=O)CC1(OCC)CN(C(C2SCC=C2C)=O)C1)CC 46566,C(=O)(CC(C)(C)C(=O)NC1CN(C(c2cn(C(F)F)cn2)=O)C1)OC 46567,c1(NS(c2ccc(C)cc2)(=O)=O)ccc(C2=CCC(O)CC2)s1 46568,C1(COC)(CNC(=O)CCN(C)CCO)CCN(C(C2CCCC2C)=O)CC1 46569,CC(C)C(O)C(C)C(=O)NC1CCN(C(c2ccn3ccnc3n2)=O)C1C 46570,c1(C(N2C(C(C)NC(=O)Cc3ccno3)CCC2)=O)cc(Cl)ccc1Cl 46571,c1(C(=O)NCC(C)NC(C2(CCC)CC2)=O)cc(COCc2ccsc2)oc1C 46572,c1(C(=O)OC)ccc(F)c2c1CN(C(=O)C(=O)N(C1CCC(C)C1)C)C2 46573,c1(C(N2CCC(NCc3cn(CC(=O)NC)nn3)CC2)C)ccc(F)cc1F 46574,C1(CC)(CC)CCCN(C(=O)CC2CCN2C(c2ccc(O)cn2)=O)C1 46575,CCCC(C(=O)NC1C2CN(C(c3cnn4ncccc34)=O)CC12)C(C)C 46576,c1(C(N2CCCC(CCNC(CCC=CC)=O)C2)=O)cc(N)c(C)cc1C 46577,c1(C(=O)NCC2CCCN(C(C(C)NC(C)(C)C)=O)C2)ncc(Br)cc1F 46578,CCC(CC)C(F)C(=O)N(C)CC1COCCN1C(=O)CCc1csnn1 46579,c1(OC)ncc(C(=O)NC2CCC(N(C)C(c3cnc(CC(C)(C)C)o3)=O)C2)s1 46580,c1(C2C(C(=O)NCCCCCNC(C(C)OCC#C)=O)C2)cc(F)c(F)c(F)c1 46581,N1(C(C=C(C)C)=O)CC2CC(F)(F)CCC2(NC(c2cc(Cl)cnc2O)=O)C1 46582,c1(C(C(=O)N2CC(c3cnc[nH]3)C2)C2CCCC2)ccccc1 46583,N1(C(CN(CCC#N)C)=O)CCN(C(=O)CCS(=O)(=O)CC2CC2)C2CC12 46584,N1(C(c2c(C)cc(C)o2)=O)CC(C(N2CCCC(F)(F)C2)=O)C(F)(F)C1 46585,c1(C(N(c2ccc(CS(C)(=O)=O)cc2F)CC)=O)cc2cc(C(=O)O)sc2s1 46586,Cc1oc2c(F)c(F)c(F)c(F)c2c1C(=O)NC1CC1(C)C(F)F 46587,C1(C(=O)NC(C2CCN(C(C34CC(CO)(C3)C4)=O)CC2)C)CCC2(CC1)CC2 46588,C1(CC(=O)NC)CN(C(=O)CCSC)CCN1C(=O)CCC1CCC1 46589,c1(CC)ncccc1NC(=O)CCC1(NC(=O)CCCF)CCC1 46590,C(=O)(C1CCCc2ncccc21)NCC1(F)CN(C(C2(C)CCCC2)=O)C1 46591,c1(C(=O)NCC2C3(CCN(C(C(CC)O)=O)CC3)C2)c(C)nc2ncccn12 46592,CN1CC(C(=O)NCC23CC(NC(c4ccnc(C(N)=O)c4)=O)(CO2)C3)CC1=O 46593,N1(C(Cc2n(C)ncc2)=O)CC2CC2(C(=O)NCC(F)CO)C1 46594,CC1CCN(C(=O)CC(C)n2cccn2)C(C)C1NC(c1ccccc1Br)=O 46595,c1(C(N2CCC(N(C(C(C)NC(CC)=O)=O)C)C2)C)ccccc1Cl 46596,c1(N2CCC(C(=O)Nc3nccnc3F)C2)ncnn2cc(Br)cc12 46597,C1(C)(CC(=O)N(CC(CNC(c2nccc(CC)c2)=O)O)C)CCS(=O)(=O)N1 46598,CCC1CC(=O)N1C.C(=O)(CCCNC)NC.C(C)(CCC)C(C)C 46599,N1(C(C2(C(C)C)CCCN2C(=O)C(C2CCCCC2)C)=O)CC2CCCC(C2)C1 46600,C1(C(=O)NC(C2(O)CCN(C(C3CCCC(C)C3)=O)C2)C)CCC2C(CC1)C2(F)F 46601,C1(NC(c2nc(CNC(c3cc(OC)nn3C)=O)oc2)=O)CCCCC1N=[N+]=[N-] 46602,c1(CC)nc[nH]c1C(=O)NCCOCCNC(=O)CCC1CCC(C(F)(F)F)O1 46603,C1(c2ccccc2)(C(=O)NC(CNC(CSCC)=O)CO)CCOC1 46604,CC1C(C(=O)NCC2(CNC(=O)CCc3nc(O)n[nH]3)CC2)=Cc2ccccc21 46605,c1(COC)cc(C(=O)NC2CC2CNC(c2cncnc2)=O)cs1 46606,c1(C(=O)NCC2C(NC(C3C(C)C3)=O)CCCC2)c(F)ccc2nc[nH]c12 46607,C1(CNC(c2n(CCOC)ncc2)=O)CCN(C(=O)CCN2CCC2)CC1(F)F 46608,N1(C(C2CCC(CC)CC2)=O)CC(CC(=O)NCCc2cncn2C)CC1(C)C 46609,N1(C(c2nc(CC)oc2)=O)CCOC(C(N2CCC(CN(C)C)CC2)=O)C1 46610,c1(C(=O)NCCCCCNC(C2C(C)(C(F)F)C2)=O)ccnc(P(C)(C)=O)c1 46611,C1(CNC(CSCCC(C)C)=O)CCN(C(C23COC(CF)(C2)C3)=O)C1(C)C 46612,Cc1cc(CC(N2CCC(C)(CCNC(C3CCS(=O)(=O)N3)=O)C2)=O)n(C)n1 46613,N1(C(C(C(C)C)C)=O)CCC2(NC(=O)CSc3nncn3C(C)(C)C)CCCC12 46614,C12(C)CCN(CC1)C2=O.C1(C(C)(C)C)CCCN(c2ncc(I)cn2)C1 46615,C(=O)(N1CCC(C(=O)NCC2CCN(C)C2)O1)c1n(CC)ncc1 46616,c1(C(=O)NC(C2CN(C(c3nccnc3Cl)=O)C2)C)cncc(C2CC2)c1 46617,N1(C(CC=C=C)=O)CCCCCC1C(=O)N(C)CC1CCCN1C 46618,S(=O)(=O)(c1c[nH]c2cc(F)ccc12)Nc1c(C)ccc(-n2cnnn2)c1 46619,c1(C(=O)NCC(C(C)C)NC(c2[nH]nc(OC)c2Cl)=O)c(S(C)(=O)=O)cnn1C 46620,n1(CC(=O)NCC2N(C(CCCCC=C)=O)C3C(C2)C3)ncn2nccc2c1=O 46621,C(=O)(C(O)CCNC(=O)CN1CC2CC2C1)NCCCNC(N)=O 46622,c1(C(N2CCC(C(CNC(C(C)(C)F)=O)O)CC2)=O)c[nH]cc(Cl)c1=O 46623,c1(C(C(=O)NC(C)(C)CC)N(C2C3CCCC23)CC)cc(C)nnc1C 46624,N1(C(C2(C)CC(=C)C2)=O)CC2C=CC1C(C(=O)NCC1(C=C)CCC1)C2 46625,c1(C(=O)NC2CC(C)(COC)N(C(c3[nH]nnc3C)=O)C2)ccn2ncnc2c1 46626,c1(N(CCCNC(=O)NC2(CSC)CC2)C)ccccc1 46627,N#Cc1ccccc1C1CCN(C(c2cc(C(F)F)on2)C(=O)NCC(F)F)C1 46628,Cc1ccn(CC(=O)NCC2CC2NC(=O)COc2c(C)occc2=O)c(=O)c1 46629,N1(C(CCCc2ccc(C)s2)=O)CC2CC(C1)CN(C(=O)C(C)C(C)O)C2 46630,C(=O)(C(C)(CC)CO)NCCC1N(C(c2cnc(CC)s2)=O)CCOC1 46631,C(CS(=O)(=O)CC(=O)NC(C(=O)Nc1cncc(Cl)c1)C1CCOC1)OC 46632,N1(c2nccc(C#N)n2)CC2(CCCC2NC(=O)CN2CC3CCC2C3)C1 46633,CC(O)(C(=O)NCC1(NC(c2cnn(CC3CCCO3)c2)=O)CCC1)C1CCC1 46634,C1(NC(c2n[nH]c(C)c2Cl)=O)CCC2(CC1)CCN(C(c1ccc(CO)s1)=O)C2 46635,c1(C(=O)NCCC2(C(N(CCCCC)C)=O)CCCC2)nc(=N)cc[nH]1 46636,c1(C(N(C(C)CNC(c2ccc(-c3cccs3)[nH]2)=O)C)=O)ncc(F)cc1N 46637,C1(C(N(C)CC2CCN(C(=O)CCc3ccccc3)C2)=O)CCC(F)(F)CO1 46638,c1(C(N2CC(NC(c3cc(CC)no3)=O)C(C)C2)=O)c(C)nc2sc(C)nn12 46639,O=C(C1CCc2ccccc21)N1CC2CC1CN2C(c1cc(F)cc(F)c1F)=O 46640,C(CCCCCCCO)=CC(=O)NCC1(OC)CCN(C(C2(CF)CCC2)=O)C1 46641,N1(C(C(C)c2cccs2)=O)CCC(O)CC1C(N1CCC(c2ccco2)C1)=O 46642,C1(C(=O)NCC2(NC(C(CCC)F)=O)CCOCC2)CN2CCC1CC2 46643,N1(CCN(C)C(c2ccnn2C)=O)CCN(C(C2CC(F)(F)C2)=O)CC1 46644,N1(C(COC2CC(NC(C(C)OC(C)(C)C)=O)C2)=O)CC2CN(C)CC2(C)C1 46645,CC(CNC(=O)CCc1cscn1)(CO)NC(=O)Cn1cccn1 46646,c1(C(=O)NCC(CNC(C(CC)N(C)C)=O)(C)O)cc(N)c(C)c([N+](=O)[O-])c1 46647,Cc1oc(C(N2CCOCC2CNC(=O)CC2=CCOCC2)=O)cc1S(N)(=O)=O 46648,c1(C(=O)Nc2c(C(=O)OC)nn(CC(F)(F)F)c2)c(C)cc(C)nc1Cl 46649,C=CCCCCC(=O)NC1CC12CCN(C(=O)C(O)CSC)C2 46650,Cc1cccc(C(CNC(=O)COCCOC)NC(C2CCS2(=O)=O)=O)c1 46651,N1(c2nccc(OCC)n2)CCC(NC(C2C=CC(=O)N=N2)=O)C(F)C1 46652,c1(N(C)CC2(OC)CCOCC2)nc(=NCC#CCCO)[nH]c2cccc(F)c12 46653,NC(=O)CCC(=O)NCC1CCN1C(C12CC1C2)=O 46654,c1(C(N2CC(C(N)=O)(CNC(C(COC)OC)=O)C2)=O)cc2c(cc1N)OCO2 46655,C1(CSC)CCCN1CCNc1nocc1C(C)(C)C 46656,CCCCC(CNC(=O)CC1(NC(=O)C(C)n2ccnc2)CC1)CCC 46657,C(=O)(C1=Cc2ccccc2C1)N1CC2C(C(N3CCC4(C3)CC4(F)F)=O)(CC2)C1 46658,CCCCCS(=O)(=O)CC(=O)N(C(C)CN(C(=O)CC(C)O)C)C 46659,N1(C(c2n(C)[nH]c(=N)c2)=O)CCCC2(CCCCC2NC(=O)CNC(N)=O)C1 46660,C1(NC(c2nc(C)oc2)=O)CC1C1CCN(C(=O)C(C)CC(C)C)CC1 46661,C1(c2ncc(C)cn2)CCN(N(CC2CCCCC2)Cc2ccc(Cl)cc2)CC1 46662,C(C(=O)NCc1ccnn1C1CCCCC1)(C(=O)O)OC 46663,C1(CC(=O)NC(C(C)NC(CCCn2c(C)ncc2)=O)CO)CC2C=CC1C2 46664,CP(C)(=O)C1(O)CCN(C(c2ccccc2Cl)C(=O)NCC2CC(F)(F)C2)CC1 46665,C1(NC(Cc2c(C)n[nH]c2)=O)CC2CC1CN(C(=O)C(CO)C(F)(F)F)C2 46666,c1(CC(CC)NC(=O)CCn2cc(-c3cc[nH]n3)nn2)ccccc1Cl 46667,C(C(CNC(=O)CC1CC1CC)S(C)(=O)=O)NC(CCC)=O 46668,Cc1ccc(C)n1CC(N1CCCC1CCNC(c1cc(C(F)(F)F)cs1)=O)=O 46669,N1(C(=O)Cc2cccnc2)CC2(CCN(C(C3CCCN3C(=O)C3CC3)=O)C2)C1 46670,c1(C(N(C(c2cocc2Br)C(=O)NCCOCC)C)C)ccc2ccccc2c1 46671,C1(NC(C2COCCN(C(C3(OC)CCCC3)=O)C2)=O)CC(C)N(C)CC1C 46672,c1(OC)cccc(CNC(=O)C(O)C2CN(C(=O)C(C)(C)C#N)C2)c1 46673,N1(C(Cn2c(C)cc(C)n2)=O)CCC2C(C1)NC(=O)CN2C(=O)CC1C=CCC1 46674,C1(NC(c2cc(O)ccc2I)=O)CC2(C1)CN(Cc1ccc(I)cc1)C2 46675,C1(NC(C(C)O)=O)(CO)CN(C(=O)CC(C)n2cccc2)C1 46676,c1(CC)nc(C)oc1C(=O)NC(C)(C)C(=O)NCc1sc(C)nc1C 46677,C(=O)(C(C)(C)C(=O)N1CCCC(N(C(=O)CC2(C#N)CCC2)C)C1)N(C)C 46678,C1(N(S(=O)(=O)Cc2cc(Cl)cc(Cl)c2)C(n2cccn2)C)CCC12CCNCC2 46679,CC1CC(C(=O)NCCOCC2CCC2)CN(C(=O)CCn2cnc(=N)[nH]2)C1 46680,N1(C(c2n(CCC)ncc2)=O)CCCC(F)(C(N2CC3CC3C3CC23)=O)C1 46681,N1(C(CN2C(C)CCC2)=O)CC(O)CC1CNC(C1COC1)=O 46682,C(=O)(C(F)C(C)(C)O)NCC(C)CC(=O)Nc1cccc(C2CC2)c1 46683,c1(C(=O)NC(CNC(CC2(OCC)CC2)=O)CC(F)(F)F)ncnc2sccc12 46684,Cc1cnc(Cl)[nH]c1=NC(=O)c1cnc2n[nH]c(-c3ccnc(F)c3F)c2c1 46685,c1(C(=O)NC2C(NC(c3cn(C)nc3C3CCCC3)=O)C2)c(N)cc(Cl)cc1F 46686,C(C(C)C)(C(O)C(=O)NCC1(O)CCCN(C(C2SC3C=CC2CC3)=O)C1)OC 46687,C(CC(C)C(=O)NCC(c1ccccc1F)NC(C1CCC1(F)F)=O)=CCC 46688,CCC(C)(O)CCNC(=O)C(C(C)OC)NC(=O)CN1CCC(=O)CC1 46689,c1(N(CC(CN(C(C(CC)NC(N)=O)=O)C)O)C)cc(Cl)nc(CS(C)(=O)=O)n1 46690,C1(NC(CC(=O)NCC)=O)CN(C(c2ccc(Br)s2)=O)CC2(CCC2)C1 46691,CC(C(=O)NCCOCCOCCNC(=O)CN(c1ccsc1)C)C(C)O 46692,N1(C(c2csc(C)c2N)=O)CC(C)CN(C(c2sc([N+](=O)[O-])cc2Cl)=O)CC1C 46693,c1(CC(=O)NCC2CCCCC2F)ccc(F)cc1.C12(COC)CN(C1)C2=O 46694,C1(C(=O)NC2CCC(F)(F)C2)CC(F)(F)CN1S(=O)(=O)CCBr 46695,c1(C(=O)NCC2CC2NC(c2sc(Cl)cc2Cl)=O)cn2c(n1)CCC2 46696,Cc1nc2ccnn2c(C)c1C(=O)NCC1COCC1NC(=O)CCC(F)F 46697,N(C(=NCCc1ccc2occc2c1)N1CCN(CC2CCCO2)CC1)CC=C 46698,c1(C(N2CC(C(C)C)N(C(=O)C(=O)N(C)C)CC2)=O)cnc2c(=O)[nH]ccc2c1 46699,N1(C(C(CCC)NC(C)=O)=O)CCOC2(CCCN(C(=O)C(O)C(C)(C)C)C2)C1 46700,C(C(C)CC(=O)N1CC(OC)CC1CCNC(=O)Cc1cncn1C1CC1)OC 46701,N1(C(c2n(C)nc(Br)c2)=O)CC(NC(=O)C2CC2)C2(CC2)C1 46702,CC(CCc1ccccc1F)C(=O)NCC1CCCN1C(c1c[nH]nc1Cl)=O 46703,N1(C(CC(CCC(CC)C)C)=O)CCC2(CCC(NC(=O)CC(F)F)CC2)CC1 46704,C1(C(N(CCCCNC(c2cc(COC)on2)=O)C)=O)CN(C)CCO1 46705,Cc1nn2cc(C(N3CC(CNC(c4cc(C(N)=O)no4)=O)C4CC34)=O)nc2s1 46706,N1(C(Cc2cc(C)no2)=O)CC(CNC(=O)CSCc2csc(=N)[nH]2)CCC1C 46707,C1(C(N(C(C)CC(=O)NC(C)Cc2nncn2C)C)=O)CC(C)N(C)C1 46708,N1(C(c2cnc(C(C)(C)C)[nH]2)=O)CC(CNC(=O)CCn2ccnc2)C(O)C1 46709,c1(C(=O)NC(CCOC)C(=O)N(C2CCN(C)C2=O)C)cccc(F)c1C 46710,c1(OC)ncc(C(N2CC(CCNC(C3CCC(C)O3)=O)C2)=O)cc1C 46711,c1(CC(=O)OCC)occc1C(=O)NC(CNC(=O)CCCNC(N)=O)C(C)C 46712,C1(CNC(c2ccc3nn[nH]c3c2)=O)CN(C(c2cc(Cl)no2)=O)CCC1(F)F 46713,N1(C(c2cnc(COC)s2)=O)CC2C(NC(=O)Cc3csc(S)n3)C2C1 46714,c1(OC)cc(C(=O)NC2CCN(C(=O)C3=C(C)CCC3)C2(C)C)c(F)c(Cl)c1 46715,CC1(C)CN(C(=O)CCC2CC2(Cl)Cl)CC(CNC(=O)C=Cc2cscn2)O1 46716,C1(N(CC#C)C(c2nocc2Cl)=O)CCN(C(C2(O)CCC2)=O)CC1 46717,N#Cc1ccc(C(O)C(=O)OCC2CCC2c2ccccc2)cc1 46718,O=S(=O)(c1ccc(Br)cc1NC1CCCn2ccnc21)N1CC2CCC1CC2 46719,N1(C(C2C(C)(NC(Cc3nc(C)oc3)=O)CCCC2)=O)CCCC(C2CC2)CC1 46720,c1(C(=O)NCCN(C(=O)COC2CCC2)CCC)snnc1CC1CC1 46721,c1(C(N(CCNC(c2cccc(N(C)C)c2)=O)CC)=O)ccc2nc(S)[nH]c2c1 46722,c1(C(=O)NC(COCC)C(=O)NCCC2CCC(C)C2)cc(OC)cnn1 46723,N1(C(CNC=O)=O)CCOC2CN(C(C3C4CC5C(C4)C35)=O)CC12 46724,CC1=C(C(=O)N2CCC(NC(=O)C(C)OC3CC3)C(F)C2)CCCC1 46725,N1(C(Cc2nc(C)sc2C)=O)CCCC(NC(C23CC(C2)C(C)O3)=O)CC1 46726,N1(C(C2(CC(C)C)CCC2)=O)CC2CCC(NC(C34CC(C3)C4)=O)C2C1 46727,C(=O)(C(C(C)C)OCC)NC.C1(=O)CC=CCOC(=O)CN1CC=C 46728,N#CC1(C(=O)NC2CCCCCN(C(c3cccnc3)=O)C2)CC12CCOCC2 46729,c1(Nc2n(CC#C)cnc2-c2ccc(F)cc2)c(OC)ncc(Br)c1C 46730,N1(C(CCc2c(C)ncs2)=O)CC=C(CCNC(=O)CCCOC(=O)N(C)C)CC1 46731,C(=O)(CC1COc2cc(O)ccc21)NC(CN(C(=O)CCCC1CC1)C)(C)C 46732,C(=O)(C1=CCC(NC(C2CCCC(=O)CC2)=O)C1)N(C(C)CO)CC 46733,c1(OC(C(=O)NCC2(F)CN(C(C=C(CCC)C)=O)C2)C)ccc(Cl)cc1Cl 46734,CC1CCC(C(=O)NCc2nc(CNC(=O)C=Cc3ncc[nH]3)cs2)C1 46735,C1(NC2(c3n(C(C)C)nnn3)CCN(CC(F)(F)F)CC2)CN2CCCC2CO1 46736,C=CCC(C)(CC)C(=O)NCC1CCC1C(=O)Nc1ccc(C)cc1CO 46737,C1(O)(CNC(C2(CCCC)CCC2)=O)CC(NC(=O)C(c2nc(C)cs2)C)C1 46738,C12(CSCc3nc(C)sc3)CC1CN(C(C1(CO)CCC1)=O)C2.C1CC(=O)N1 46739,CCC(O)C(C)C(=O)N1CCCCC1CCNC(C1CCCCN1S(C)(=O)=O)=O 46740,N1(Cc2nc(CC)[nH]n2)CCC(F)(C#N)C1.C1(=O)CCCN1 46741,CCCCC(CNC(C1CCC(CN2CCOCC2)O1)=O)NC(=O)CC1CCC1 46742,CC1CCc2c(C(N3CC(NC(C4CCC(C)(O)CC4)=O)C(C)C3)=O)csc2C1 46743,Cc1cc(C(=O)N(C(CNC(c2cccc(O)n2)=O)C2CC2)C)n2nccc2n1 46744,c1(C(N2C3CC(NC(CCC#C)=O)C2CC3)=O)ccc(=O)n2c1CCC2 46745,Cc1cc(C(=O)NC2(C)CCC(NC(C3CCCS3)=O)CC2)n2nccc2n1 46746,C(=O)(C(F)(F)C(C)O)NC1CC(NC(C2(OC(C)C)CCC2)=O)CC1O 46747,CC1CCCC(CNC(C2(NC(=O)Cn3cc(Br)cn3)CC2)=O)O1 46748,CC(C)C(O)CC(=O)NCc1ccsc1C(N1CCCC(F)(CO)C1)=O 46749,C1(N(C(=O)CCC2CCCCO2)CC)CCCN(C(=O)CSc2nncs2)CC1 46750,CC1CC(NC(=O)CCS(N)(=O)=O)CCN1C(C1CC2(C1)CC2(F)F)=O 46751,C(=O)(C(C)CCCc1ccccc1)N(CCNC(C=CCCC=C(C)C)=O)C 46752,c1(CC)cc(C(=O)NCC=CCNC(=O)C(F)(F)c2ccnn2C)oc1CC 46753,Clc1ccccc1-n1ccnc1Cn1ccnc1C1COCCO1 46754,Cc1cc(=NC(C)CN(C(=O)C2=NOC(C3CC3)C2)C)[nH]c(C2CCCCC2)n1 46755,N1(C(C2C(C)(C)CCCC2)=O)CC2COCCC2(NC(=O)Cc2cc[nH]n2)C1 46756,C1(C(=O)NCC(C2CCN(C(c3cnc[nH]c3=N)=O)CC2)C)CCCCC12CC2 46757,c1(C(N2CC(NC(C=CCOCCOC)=O)C(O)C2)=O)cccc2cnsc12 46758,c1(C(N(C2(C(=O)NC3(CO)CCCC3(C)C)CC2)C)=O)cc2ccccc2[nH]1 46759,c1(C(=O)NCC(C)(CC)NC(CCC#CC)=O)cc2ccccc2nc1C(F)F 46760,C1(C(C)(C)NC(C2C(=C)C2)=O)CCN(C(C2CCOC(=O)N2)=O)CC1 46761,C1(C(N(CC2OCC(=O)NC2)CC2(C(F)(F)F)CC2)=O)CCC2(CCNC2)CC1 46762,c1(C(C(=O)NCC=C)N(CC(=O)NCc2cccnc2)C)cn(C)cn1 46763,CCC(CC(=O)NCC1CCN(C(=O)CC2CN(C(C)=O)C2)CC1)C1CC1 46764,CC1OCCC1CC(=O)NOCC(=O)NCC1(CCCO)CC1 46765,C1(C2(O)CCOC2)(CNC(c2n(C)c(O)nc2)=O)CCC1 46766,C=CCCC(F)(F)C(=O)NC1CN(C(=O)Cn2cnnc2O)CC2(CC2)C1 46767,C1(NC(c2cc(SCC)ncc2)=O)CC2CN(C(=O)C=CCO)CC12 46768,CC1=NOC(=O)C1CC(=O)NC1CCC(NC(=O)CSc2nncn2C2CC2)C1 46769,O(P(=O)(OCC)C1(C)CCCN1C(=O)Nc1nc2ccc(C(F)F)cc2s1)CC 46770,CCC(CN(C)C)CC(=O)N(C)CC1(O)CCN(C(c2cncn2C(C)C)=O)C1 46771,N1(C(CC2(CC=C)CCCC2)=O)CCC2CCN(C(C3C=CCC3)=O)C2C1 46772,c1(NC(C2CSCCN2Cc2scc(Br)c2Br)=O)ccc(O)cc1Br 46773,c1(C(N2C(C)CC(CNC(C3COCCO3)=O)C2)=O)ccc2c(c1)CCN2 46774,C1(NC(c2c(C)n[nH]c2)=O)COCCN(Cc2ccc(Br)cn2)C1 46775,c1(C(N(C)CC2CCN(C(c3coc(C(F)F)c3)=O)C2)=O)ccc2c(c1)COC2 46776,N1(C(c2nnn(C(C)(C)C)n2)=O)CCCC(C)(NC(=O)CC2CCC(=O)N2)C1 46777,c1(OC)ccc(C(=O)NC2CCCC2NC(=O)C(O)CC(F)F)cc1OC(F)F 46778,N1(C(C2(C#C)CCCC2)=O)CC2CCOCC2(NC(=O)CC(C)(C)CC)C1 46779,c1(OC)ncnc(N2CC3CC2C3C(N2CCC(C)(O)C2)=O)c1C 46780,c1(CC(=O)N(CC(CN(C(C2C(=C)C2)=O)C)O)C)cc(Br)nn1C 46781,C1(NC(C2(C(C)C)COC2)=O)CC(CNC(=O)C(C)CC2CC2)CC1O 46782,N1(C(C(CC)=CC)=O)CC(OC)C(NC(=O)CC2(CO)CC2)C1 46783,C1(C(C)C)CN(C(=O)CC(C)(C)C(F)F)CCCN1C(=O)CCCCC1CC1 46784,N1(C(c2c(CC)occ2)=O)CCOCC(CNC(=O)C=Cc2cn[nH]c2)C1 46785,C1(C(=O)NC2CC3(OCCC(N)C3)C2)CCC2(CCCCC2)CC1 46786,CC1CCCC1C(=O)NCC(C)(C)CN(C(=O)Cc1cnc(C2CC2)[nH]1)C 46787,c1(C(=O)NCC#CCNC(CN(CCC#C)C)=O)csc(O)n1 46788,Cc1ccc2cc(Cl)cc(C(=O)NCCn3cc(-c4csc(C)n4)nn3)c2n1 46789,c1(NCCNC(C2=NN(CC)C(=O)CC2)=O)cc([N+](=O)[O-])c(N(C)C)cc1F 46790,C12(C(=O)NC3CC(CCNC(C4(OC)CCCCC4)=O)C3)CCC(C)(CO1)C2 46791,C1(C(=O)NC(C(N2CCC(c3ncco3)C2)=O)c2cccs2)CC=CC(O)C1 46792,c1(CCOC)ccc(N(C(c2ccc(CC3CC3)cc2)C(=O)NC(C)C)C)cc1 46793,N1(C(C(C=C)(C)C)=O)CCC2(CCCN2C(C2CCC3(CCOC3)O2)=O)CC1 46794,c1(NC)ccc(C(=O)NC2(CCCC(=O)N3CCC(C(N)=O)C3)CCC2)cc1 46795,C(=O)(CC(C)C(C)(C)NC(=O)Cc1ccccc1O)N1CC(CC)N(C)CC1 46796,c1(C(=O)NC2C(NC(C3N(C)CCCC3)=O)CCCC2)cccc(=S)n1O 46797,c1(C(=O)OC)cc(-c2cc(CN)nn2C)cn(C)c1=O 46798,c1(C(C)OC)ncc(C(=O)NCCN(C(=O)C(C)(C)F)C(C)C)s1 46799,C1(NC(c2cccc(SC)c2)=O)CC2(NC(c3c(Cl)n[nH]c3C)=O)COC1C2 46800,C(C(=O)N1CCC(NC(C2CC2F)=O)C1)(C(C)(C)C)NC(=O)OC 46801,N(C1CCCc2c[nH]nc21)C(C(C1CC1)NC(c1cn[nH]c1)=O)=O 46802,C(CC(C(=O)NC(CC1CC1)CC1CC1)NC(=O)CCC1CCC(=O)C1)OCC 46803,C12(C(=O)NC3(CC=C)CCN(C(C4(C)C(C)(C)C4(C)C)=O)C3)CCCC1C2(F)F 46804,C(=O)(CC(C)CCCCC)N1CCC(N(C(=O)CC(C)(C)COC)CC#C)C1 46805,C(C(=O)NCCC1CCN(C(=O)CNc2nccs2)C1)(C(C)C)N(CC)CC 46806,O=C(CC(F)(F)F)NCC1CCCCC1NC(c1ccc(OC(F)(F)Cl)cc1)=O 46807,N1(C(C(C2CCC2)OC)=O)CCC12CN(C(=O)CCCSc1ccccc1)C2 46808,c1(C(N2CCCC(CN(C(C3C(C)C3)=O)C)C2)=O)ccc(F)c2occc12 46809,C(=O)(C1CCCc2ncccc21)N1CCC(CCCNC(C(C)SCC)=O)CC1 46810,C(=O)(C(F)(F)C(C)O)NC1CC(CCNC(c2ccc(CCC)[nH]2)=O)C1 46811,c1(C(N2CCN(C(C3CCC(=O)NC3)=O)CC2CO)=O)coc2c1CCCC2 46812,CC1CN(C(=O)CC2(C)CCOCC2)CC(C(=O)NCC2(CO)CC23CCC3)O1 46813,C1(Cc2ccc(OC)cc2)CCCCNC1=O.C12(O)CCN(C1)C(C)CNC2=O 46814,c1(C(=O)NC(C(C)C)CCNC(=O)CCCN(C)C)ccc2c(c1)C=CCC2 46815,C1(C)(C(N2CCC(CN(C)C(c3cccnc3O)=O)C2)=O)COCCO1 46816,c1(C(=O)NC(CNC(C(CC)c2ccccc2)=O)C2CC2)[nH]c(C)nc1C 46817,N1(C(C(COC(C)C)(C)C)=O)CCC2(CC2NC(c2ncoc2C2CC2)=O)C1 46818,C(=O)(C(C)CCCOC)NC1C(CC)CN(C(c2cnn(C3CCC3)c2C)=O)C1 46819,C(CC(C)(C)C)N(CC(=O)NCC1CCCN1C(=O)CCC1CCOCC1)C 46820,c1(CC(N2CCC(OCC(=O)NC3CCC3CO)C2)=O)cccc(F)c1 46821,CC1CC(N(C)C(C2C(C)CN2C(C2CCN2C(C)(C)C)=O)=O)CCO1 46822,c1(C(N2C(C)CC(NC(C3CC3(C)C)=O)CC2)=O)cc(F)c(O)c(F)c1 46823,c1(NC(C2C(CNC(c3c[nH]nc3Cl)=O)CC2)=O)ccc2n[nH]cc2c1 46824,C1(NC(C23CCC(NC(c4c(CC)n[nH]c4)=O)(CC2)C3)=O)CCN2CCCCC12 46825,C#CCCCC(c1ccc(Br)cc1)NC(c1cc(-c2ccc(F)cc2)n(C)n1)=O 46826,c1(C(=O)NC2CCN(C(c3cnc(-c4ccoc4)s3)=O)CC2)cnn2c1OCC2 46827,c1(NC(=O)NCCCC(N2CCc3nc[nH]c3C2)=O)cc(F)c(Br)cc1F 46828,C1(CC)CCC(C)CN1C(=O)COC1CCN(C(c2ccoc2Cl)=O)C1 46829,CCC(CC(=O)N1CCCC1CNC(c1cc(C)nnc1O)=O)C(C)C 46830,c1(C(=O)NC(c2ccc(CNC(COC)=O)cc2)C)ccc(Br)nc1N 46831,c1(C(=O)NC2CCN(C(C(CCC)OC)=O)CC2(C)C)cc2c(C)cccn2n1 46832,C1(NC(Cc2cc(C)ns2)=O)CN(C(=O)C(C)Sc2nncn2C)CC1C 46833,C1(N(C(=O)CC2COC(=O)C2)C)CCN(C(c2cnc[nH]2)=O)CC1 46834,c1(C(N(C(CNC(C(C2CCOC2)OC)=O)C2CC2)C)=O)cn2cccnc2n1 46835,N1(C(CC=C=C)=O)CC2(CCOCC2)CC1CNC(c1cnc2sc(C)cn12)=O 46836,c1(C)ccccc1SC.C(CCCCC(=O)NOC(C)CC)SC.C1(C)C(=O)N1 46837,C1(C)(NC(CC2(C)N(C(c3ccc(C(C)C)o3)=O)CC2)=O)CCCC1C 46838,C1(NC(C(CC)COC)=O)CN(C(c2cnc(OC)nc2)=O)CC1S(C)(=O)=O 46839,c1(CCC(=O)N(C2CCCN(C(C3CCOC3)=O)C2)C)cn2ccccc2n1 46840,C1(CNC(CC2(C(=O)OC)CC2)=O)CC(OC)CN1C(c1ccncn1)=O 46841,C1(NC(Cn2cc(CN(C)C)nn2)=O)COCCN(C(C2CCCCC2O)=O)C1 46842,N1(C(COCC(C)C)=O)CCC(CNC(c2sccc2CO)=O)C(O)C1 46843,Cc1cc(C(=O)NC2CCCCC2NC(=O)C(c2ccc(Cl)cc2)O)nnc1C 46844,CCCCC(CC)C(=O)NCCOCCCN(C)C(C12CC(C(F)F)(CO1)C2)=O 46845,C1(NC(c2cc(C)c(Br)o2)=O)CN(C(=O)CN(C)S(N)(=O)=O)CC1C1CC1 46846,N1(C(c2n(CC#C)ccc2)=O)CCN(C(C2CCCS(=O)(=O)C2)=O)C(C(C)C)C1 46847,Cc1nc(C(=O)NC2CCC2NC(c2csc(Cl)c2)=O)c(C)s1 46848,C#CC1(C)COCCN1C(c1cnn2c1CCC2)C(=O)NCC1CCOCC1 46849,N1(C(c2n(C)nc([N+](=O)[O-])c2)=O)CCCC2(CCCCC2NC(=O)CO)C1 46850,CN1CCCC(C(=O)NC(C2CCN(C(c3ccoc3)=O)CC2)(C)C)C1 46851,C1(CC(N2CC=CC(NC(c3c(C)cco3)=O)C2)=O)CCCC(F)(F)C1 46852,CC1=CC(C)C(c2cn(CC3CN(C(=O)CNC(=O)CNC(C)=O)C3)nn2)CC1 46853,C1(C(N2C(C)CC(CNC(CCC(C)N(C)C)=O)C2)=O)CC2(CCO1)CC2 46854,C1(CNC(c2c(COC)scc2)=O)CCC2(CCN(C(=O)C(C)C#N)CC2)CO1 46855,CC1CN(C(=O)C(Cn2cncn2)NC(=O)CC2CSCCO2)CCS1=O 46856,C1(O)(CNC(c2ccn(CCOC)n2)=O)CCCN(C(=O)C(C)NC(C)=O)C1 46857,C1(C(N(CCN(C)C)C)=O)CCC(n2cc(CCC3CC(O)C3(C)C)nn2)CC1 46858,c1(C(=O)NCCCOCCN(C)C(C2C3CCCC23)=O)cc(C(F)(F)F)[nH]n1 46859,C1(N(C(C(C2CC2)OC)=O)C)CCC(NC(c2nnsc2C(F)F)=O)CC1 46860,C1(C(N)=O)CC(C(=O)NCC(C)(C)CNC(=O)CCSc2ccccn2)=NO1 46861,c1(OC)cccc(C(=O)NC2CCN(C(C3(C#N)CCCO3)=O)C2)c1C 46862,CC1(CC(=O)NC2CC(F)(CNC(=O)COCCCF)C2)Oc2ccccc2O1 46863,Cc1cccc(C(=O)C(=O)NC2CCN(C(c3cnc(C4CC4)o3)=O)C2)c1 46864,C12(C(N3CC(O)(C(C)NC(=O)C(F)CC4CCC4)C3)=O)CC3CC1C2C3 46865,N1(C(c2n(CC)ccc2)=O)CCOC2CN(C(=O)C(c3ccccc3F)C)CC12 46866,CCC(C)C(C(=O)NCC(C)C(F)F)NC(C1CCCSC1C)=O 46867,C(CCC(C)(c1nnnn1CCCF)NC1CC1Cc1ccccc1)OCC 46868,c1(C(=O)OCC)cnc(C(C)C)[nH]c1=NCCCN(C(=O)CC(C)(F)F)C 46869,c1(C(=O)NC(CN(C(=O)C(C2CCOCC2)F)CC)C)cc(C(C)C)n(C)n1 46870,c1(C(N2C(C)(CC)CC(NC(=O)CC3=CCCC3)C2)=O)nc2c(s1)COCC2 46871,C(c1cncnc1O)=CC(N1C(C)CC(NC(C2N(CC#C)CCC2)=O)C1)=O 46872,CC(C)C#CC(=O)NCC1(C(N)=O)CN(C(C2CC(O)C(F)C2)=O)C1 46873,C1(C)(C(=O)NCC(N(C(C(C)n2cccc2)=O)C)C2CC2)CCCS1(=O)=O 46874,C12(CCNC(=O)Cc3ccccc3F)CCC(C1)N(C(c1ns[nH]c1=O)=O)C2 46875,C1(CC(C)NC(C2(CC#C)CCC2)=O)CCN(C(=O)CNC(C)=O)CC1 46876,C12(C(N3CC(SC)C(NC(=O)CC4CCCN(C)C4)C3)=O)CCC(CC1)CC2 46877,C1(C(N2CC(O)(CNC(Cc3cc(OC)no3)=O)C2)=O)Cc2cc(C)ccc2O1 46878,c1(C(=O)NC(C)CCF)ccc(CNC(C2CC2F)=O)nc1 46879,C1(NC(CCSCCC)=O)CC(C)N(C(=O)C(=O)NCC(F)F)C1 46880,C12(NC(CCCC#C)=O)CCN(C(c3cnoc3-c3cnn(C)c3)=O)CCC1C2 46881,C(=O)(C1OC(=O)c2ccccc21)N1CC(NC(CCC)=O)C(C)(C)CC1 46882,CCCC(CNC(=O)C(CC)OC)C(=O)NC1CCN(CCC)C1 46883,c1(C(=O)NC(CC)CN(C(=O)C=Cc2scnc2C)C)ccc(CO)cc1OC 46884,C(CC(C(N)=O)NC1CCSC1)OC 46885,C1(NC(C(=O)N(C)C)=O)CC2CCC1N(C(c1ccccc1Cl)=O)C2 46886,c1(C(C)(C)C)ocnc1C(=O)NCC(C)(C1CCC1)NC(=O)Cn1cnnc1O 46887,N1(C(C2N(CC)C(=O)CC2)=O)CCCC(NC(c2cnc(C)n2C)=O)C1C 46888,C1(C)(NC(C2(F)CCN(C(C(C)SC(C)C)=O)CC2)=O)CCCCC1(C)C 46889,S(=O)(=O)(c1sc(O)nc1C)N(C1CC2CC1CC2(O)c1ccccc1)CC 46890,C=C(Cl)CC(C(=O)NCc1cnc(F)c(C)c1)NC(=O)C(C)C(F)(F)F 46891,c1(NC(COC)CC(C)C)cc(N(CC(C)CO)C)nc(C)n1 46892,NC(=O)C(N)CCC(=O)NCC1CN(C(c2ccc(C3CC3)nc2)=O)CCO1 46893,CC1CCN(C(C2(CCF)CCC2)=O)CC1CNC(=O)CCC(C)(C)F 46894,c1(C(=O)NC(C2CN(C(c3cnn(C4CCCCC4)c3)=O)C2)C)ccsc1C#N 46895,Cc1c(C(N2CCC(NC(c3cncc(Cl)c3)=O)C2C)=O)ccn1CCO 46896,C(c1ccc(OC(F)(F)F)c(O)c1)=CC(N1CCN(c2ccc(Cl)cc2)CC1)=O 46897,CCC(C(=O)OC)C(=O)N1CCCCC1CN(C)C(c1sc(OC)nc1Cl)=O 46898,c1(SCC(=O)NCCCN(C(CCCC#C)=O)CC)ccc(Br)cc1C 46899,Cc1csc2ncc(C(=O)NC3CN(C(=O)CSC(F)(F)F)CC3O)n12 46900,Cn1cc(Br)c(=NC(=O)CCN(C2(O)CCC2)C(=O)OC(C)(C)C)[nH]1 46901,c1(CCC)nc(C)c(C(N2CC(CNC(C3(C#N)CCC3)=O)CC2C)=O)o1 46902,C1(OC)CC(C)N(C(=O)C(=O)NCCCc2nn[nH]n2)C(C)C1 46903,c1(C(=O)NC(CN(C(C2(COC)CCCO2)=O)C)C)cc(Cl)c(N)cc1OC 46904,C#CCC(C)(C(=O)NC(C)C(=O)OCC)NC(=O)CN1C(=O)CNC1=O 46905,N1(C(c2n(C)c(S)nn2)=O)CCCN(C(c2ccc(N)cn2)=O)CC1 46906,C1(C(=O)NCC(C)(CO)NC(=O)CN2CC3CC3C2)CCC(=O)NC1 46907,N1(C(COC(C)C)=O)CCCC2CN(C(=O)CN3CCN(C)CC3)CCC12 46908,N1(C(C(CC)(C)C)=O)CCC2CN(C(c3c(OC)ccnc3F)=O)CCC2C1 46909,C(CC(C)C)(C(=O)N(C1CC1C)C)N(C(CC1(OC)CCCC1)=O)C 46910,n1(CC)nc(C(N2CC(NC(=O)CCc3ncccn3)CC2C)=O)cc1O 46911,N1(C(C2C(C)CCO2)=O)CC2CC1C2NC(=O)COCC(N1CCCC1)C 46912,c1(C(=O)Nc2cc(C(C)C)[nH]n2)nn(C)c(NC(C2(CC)CC2)=O)c1Cl 46913,Cc1nc2ccnn2cc1C(N1CC(NC(=O)C=CCF)C(C)C1)=O 46914,c1(C(=O)NCCCCCN(C)C(C23CC(C)(CO2)C3)=O)cc(Cl)cnc1O 46915,c1(C(=O)NCC2(F)CC(CNC(c3sc(CC)c(C)c3)=O)C2)cc(N)cc(F)c1 46916,c1(N2CCC(O)(C(C)NC(c3cncc(Cl)c3)=O)C2)ncc2c(n1)CCCCC2 46917,N1(C(C(=O)NC(CC)C)CC2C=CCC2)CCC(CS(C)(=O)=O)CC1 46918,C1(NC(=O)CCCn2ccccc2=O)CN(C(=O)Cn2nccn2)CCC1CO 46919,c1(C(=O)NC2CN(C(CSc3ccc(OC)cc3)=O)C2)nc2cccnc2s1 46920,C(=O)(C(O)CCCNC(=O)CC1CCOC1(C)C)NCC1CC(SC)C1 46921,S(=O)(=O)(c1cccc(Cl)c1Cl)N1CC2(CC(CC(=O)Nc3cc(I)ncn3)C2)C1 46922,Cc1c(C(=O)N(CC(C)NC(=O)CCC=CBr)C)ccn1C 46923,N1(C(C=CCN(C(C(c2ccn(C)n2)C)=O)C)=O)CCOC(C2(C)CC2)C1 46924,c1(CC)ncc(C(=O)NCCOC2CCN(C(C3CC3C(C)(F)F)=O)C2)c(O)n1 46925,c1(C(=O)NC2CCN(C(C(F)=CC)=O)CC2(C)C)cc2c(nc1O)CCCC2O 46926,Cc1nnc(N(C2CNC2)C(C2(C)CCCC2(F)F)=O)nc1C 46927,c1(NC(c2n(CCC)nnn2)CCc2ccccc2)cc(COC)ccc1OC 46928,N1(C(CC2(CC=C)CCCC2)=O)C2CCC1C(CNC(c1cc(C)ns1)=O)C2 46929,c1(NCC)cc(C(=O)NCCC2CC2)on1.C(=O)(COCCOCCO)N 46930,c1(C(N2CC(NC(C(C)(F)c3ccccc3)=O)C(O)C2)=O)cccc(Cl)c1Cl 46931,CCCC(C(=O)NCC(CO)NC(c1c[nH]nc1CC)=O)OC 46932,CCCCC(O)C(C)C(=O)N(CC(=O)NCC1CC2C=CC1O2)C 46933,c1(C(=O)NCC2C(NC(=O)CCN3CCCC3)CC2)cnc(C(F)(F)F)c(F)c1 46934,N1(C(C2CCC(=C)CC2)=O)CCCC(C)(NC(=O)CC2CCC2(F)F)C1 46935,c1(C(=O)NC2(C(N3C(CC(C)(C)C)CC3)=O)CC2(C)C)cnn2c1CCC2 46936,C=CCCC(=O)NCCC(C)N(C)C(c1occc1Cl)=O 46937,c1(OCC)ccc(C2CCN(C(=O)C(N3CCOC(CN(C)C)C3)=O)C2)cc1 46938,C(=O)(C(F)CCCCC(CC)CC)NC1CC2(CC(C(=O)OC)C2)OCC1 46939,c1(CNC(c2cccc(N)c2F)=O)nc2c(s1)CCN(C(=O)CNC(N)=O)C2 46940,C1(C(=O)NCC2(CNC(C(C=C)O)=O)CCC2)CCC2(CC1)CNC(=O)C2 46941,c1(C(=O)NC2CCN(CCNC(CCC)=O)CC2)c[nH]c2c(Cl)cccc12 46942,C1(C2CCC2)(CNC(C2C(=C)CC2)=O)CCN(C(c2cnc(O)c(C)c2)=O)CC1 46943,C1(CNC(c2ncn(C)c2)=O)C2CN(C(c3ccccc3C3CC3)=O)CC12 46944,C#CCC(C)(C(=O)NC(C(F)(F)F)C1CC1)NC(C1COCOC1)=O 46945,c1(C(=O)NC(CCCNC(c2cc(OC)c(C)cc2)=O)C)cc2n(c1)CCCC2 46946,CC(CC1=CCCCC1)(C(=O)O)NC(=O)COCCn1cc(CNCCO)nn1 46947,CCCC(CCCNC(=O)Cc1nonc1C)NC(c1c(C)nn(CC)c1C)=O 46948,N(C(=NCC(C)OC(C)(C)C)NC1C(C)(C)C1(C)C)C(CC)C 46949,c1(N2CC3OCC(COC)C3C2)nc(=NC)[nH]c(=NCCCC(=O)NC(C)C)[nH]1 46950,C(=O)(CCC(=O)c1cnn(C)c1)N(CCCNC(c1c(COC)cco1)=O)C 46951,C1(NC(CC=CCC)=O)COC2(CCN(C(C3(CO)COC3)=O)C2)C1 46952,C12(CNC(C(F)(F)C3(OC)CCC3)=O)CCC(NC(C3CCCN3C)=O)(CO1)C2 46953,C(CC(=O)N1CC2CC1CN2C(=O)CC(C)(C)C(F)F)(C(F)(F)F)OC 46954,c1(SC)cc(C(N2CC(N(C)C(c3cc(C#N)cs3)=O)C2)=O)ccc1[N+](=O)[O-] 46955,C=CC(C)(CC)C(=O)N1CCCC1C(=O)NC1CCOC(C)(C)C1 46956,c1(N(C)C)cccc(CNC(c2ccn(C3CCNCC3)n2)=O)c1 46957,c1(C(C)=O)cc(C(=O)NCC2CN(C(c3ccon3)=O)CCCO2)c(C)nc1C 46958,N1(C(Cc2c(C)non2)=O)CC(C)(C)CC1CNC(C1CCC1(C)C)=O 46959,CCCCCCCCC(=O)NC(C)(C)CC=CC(=O)N(CC(C)CO)C 46960,C1(NC(CS(=O)(=O)NCC)=O)CCCC12CN(C(=O)C=Cc1ncc(C)[nH]1)C2 46961,C(=O)(C1=NNC(=O)CC1)N1C(C)CCC(NC(c2cc(SC)oc2)=O)C1 46962,C(=O)(C1=CCC(C)(C)CC1)NCC1CCC(CNC(c2ncn(CC)n2)=O)CC1 46963,c1(NC(C2N(C(c3cc(CC)[nH]n3)=O)CC(O)C2)=O)ncc(Br)nc1C#N 46964,C=C(C)C(CC(=O)NCCC(C)N(C)C(c1cc(F)c[nH]1)=O)OCC 46965,C(CCCO)N(C(C)C)C(C1CC1C(C)NC(C1CC1C)=O)=O 46966,c1(CC)ccc(O)c(C(=O)NC23CC(CNC(c4c(C)coc4CC)=O)(C2)C3)c1 46967,C#Cc1ccc(Br)c(C(=O)NCC2CN(C(c3cc(C)oc3C)=O)CCO2)c1 46968,C1(NCc2c(SCC)cccc2)CCCCC1(C)C(=O)OCC1CCC1 46969,C(=O)(C(C(=O)NC(C)(CNC(=O)C(=Cc1cn[nH]c1)C)CO)OC)OC 46970,C(C(O)(C(F)(F)F)c1ncc(C)o1)NC(=O)NC1CN(C(CC(=O)OCC)=O)C1 46971,C(=O)(C(F)C(CC)CC)N1C(C(=O)NCC2(C=C)CCOCC2)(CC)CCC1 46972,C(=O)(C1OC(=O)c2ccccc21)NCCCNC(CSC(=N)N)=O 46973,N1(C(c2cn(CCOC)nn2)=O)CCC(C)(NC(=O)C(F)CC2CC2)CC1 46974,N1(C(C2(F)CC2)=O)CC2CCC(C1)N2C(C1C2CC2C2CC12)=O 46975,c1(C(C(=O)N(CCCN(C(Cc2c(C)cc(C)s2)=O)C)C)O)ccc(Cl)c(Cl)c1 46976,C1(=CCNC(C(C)CO)=O)CCN(C(=O)CN(C)Cc2ccccc2)CC1 46977,C1(C(N(C)N2CCC(N(C)C)C2)=O)CCN(C)S1(=O)=O.Cc1cnc(C)cn1 46978,CCC(CC)(CC)C(=O)NCCCOCCN(C(=O)Cc1c(C)cccc1C)C 46979,N1(C(C2CN(C)C2)=O)CCn2c(-c3ccc(Cl)cc3)nnc2C1 46980,CC1CN(C(c2cn(CCO)nn2)=O)CCCN1C(=O)CC1CCCNC(=O)C1 46981,C(C1CCCn2cc(C(C)(C)C)nc21)NC(C(CC)c1nn[nH]n1)=O 46982,c1(C(C)=O)cc(C(=O)NC2CCC(CNC(=O)Cn3cc(Cl)cn3)C2)ccc1C 46983,CCCC(C(O)C(=O)NC1CCN(C)C1=O)NC(=O)C(C)C(F)F 46984,N1(C(CNS(NC)(=O)=O)=O)CCN(C(c2n[nH]cc2C(=O)OC)=O)CC(CO)C1 46985,c1(C(=O)NCC(N2C(CCC#C)CCCC2)=O)cc(C)c(Cl)c(C)c1 46986,c1(COC)cccc(CS(=O)CC(=O)NCc2ccc(C)nc2)c1 46987,c1(CNC(C2(CC)CCCCC2)=O)ccc2c(c1)CN(C(=O)CCC(C)SC)C2 46988,c1(C(N2CC(CC=C)(C(=O)NCC(C)CCCO)C2)=O)nc(C)ccc1C 46989,CCC(C)C(C)C(=O)NC(C)(C)CN1CCN(C(c2cc(OC)nn2C)=O)CC1 46990,N1(C(Cc2cc(CC)no2)=O)CC2CC2(CN2CCCC(C(=O)NC)C2)C1 46991,c1(C(=O)NC(C2CN(C(C3C(OCC)C3)=O)C2)C)nccn2ccnc12 46992,C1(N(C(CCOCCOC)=O)CCF)CCCN(C(=O)CCC2(C#N)CCC2)C1 46993,N1(CC(C)C)CCCC(C(=O)NCC(C)(C)CN(C)C(C2CCNC(=O)C2)=O)C1 46994,C(CN=[N+]=[N-])(C(=O)NCC(C)S(N)(=O)=O)NC(C(N1CC(C)C1)C)=O 46995,C(CCO)(C(F)F)N(C(=O)CNC(=O)C(O)CC1CCCC1)C.C12(C)CN(C1)C2=O 46996,C1(NC(C(C)SCc2ccccc2)=O)CCCC(NC(c2ccnnc2O)=O)C1 46997,c1(C(N(C)CC2CCCN2C(C2CCCC2(C)C)=O)=O)cc2c(s1)CCC2 46998,c1(C(N(CCNC(c2cnc(COC)s2)=O)C2CC2)=O)ccnc(S(N)(=O)=O)c1 46999,C1(C(N2CCOCC2)=O)Cc2nccnc2CN1C(=O)C1=NOCC1 47000,C(=O)(C(C)(C)CC(C)(C)C)NCCN(C(=O)Cc1csc(N2CCNC2=O)n1)C 47001,N1(C(C(C)N(C)C)=O)CCCCC1CNC(=O)CCNC(C1CC2(CC2)C1)=O 47002,C(=O)(C(CC(C)C)ONC(=O)CCC1CCOC1)N(CC(=O)NC)CC=C 47003,C(=O)(CCCCCn1cnnn1)NC1CCCN(C(c2ccc(OC)cc2)=O)C1 47004,c1(C(N(CCOC2CN(C(=O)C(O)C(C)C)C2)CC)=O)cc(P(C)(C)=O)ccn1 47005,c1(C(=O)NC2CC(N(C(C(c3cnccn3)C)=O)C)C2)occc1C1CC1 47006,N1(C(CCc2c(C)ncs2)=O)CC(NC(=O)C(C)C(C)(F)F)CC2(CC2)C1 47007,CC1CCN(C(=O)COC2CCC2)C1CNC(=O)Cc1ccc(F)cc1 47008,c1(C(=O)NCC2CC(C)(C)N(C(=O)CO)C2)cc(Br)c2nccn2c1 47009,C(=O)(CCCC(=O)N1CC2(CCNC(=O)CN(C)CCO)CCC1C2)NCC 47010,c1(COCCOC(COC(C(C)SC2OCCC2(C)C)=O)=O)ccc(F)c(F)c1 47011,c1(C(=O)NC2C(C)N(C(c3cccc(Cl)n3)=O)CC2)c(F)ccc(F)c1N 47012,C1(CNC(c2c(C)csc2)=O)C(C2CC2)CCN1C(=O)CC(C)C(F)(F)F 47013,c1(NC(C(=O)NC(C)C2CC2)=O)ccc(OCCN(C)C)cc1 47014,c1(C(=O)NCC(C)(CC)NC(C(CC)=CC)=O)cccc2c1ccn2C(C)C 47015,C1(C2CCN(C(c3ns[nH]c3=O)=O)C2)CCCCN1C(c1cscn1)=O 47016,CN(C1CN(C(=O)CCCC2CCCC2)CCc2ccccc21)C(=O)C=CCO 47017,C(=O)(C(C)(C)CC(C)(C)C)NCCC1(CNC(c2nccc(C)n2)=O)CC1 47018,CCC(N=c1cc(NCCOCC2CCCCO2)nc(SC)[nH]1)C(C)C 47019,c1(C(=O)N(C2CCC(C(F)(F)F)CC2)CCO)nc[nH]c2nccc1-2 47020,C(=O)(C(F)n1ccnc1)N(C(C)C(=O)NCCNC(N)=O)CC 47021,C1(CNC(C(=O)NC(C)C)=O)COCC2(CCN(C(=O)CCCC3CC3)C2)O1 47022,N1(C(C2(CCN=[N+]=[N-])CC2)=O)CC(=O)NCC1C(N1CCNC(=O)C1)=O 47023,c1(C(=O)NC(CC(C)NC(c2c(NC)cccc2)=O)C)c(F)cc(C)cc1Cl 47024,C(C)(C(C)C(=O)NCC1(C2CCC2)CC1)NC(C(C=C)C)=O 47025,c1(C(=O)NCC#CC)c[nH]nc1CCNC(C1CCN1C(C)(C)C)=O 47026,N1(CC)CC(NC(=O)Cn2cc(CNC(c3nc(C)c(C)s3)=O)nn2)C(C)C1 47027,C1(NC(c2cc(CC)[nH]n2)=O)CCCCN(C(c2cnc(C)cc2Cl)=O)C1 47028,c1(NC(C2CC2Cl)=O)cccc(Oc2cccc(Br)c2)c1 47029,Cc1cn2c(n1)C(C)N(C(N1CC3(CC(CC(=O)OC(C)(C)C)C3)C1)=O)CC2 47030,c1(C(=O)NCCN(CCC)C(C)C)cnn(CCNC(=O)CCN2CCCC2)c1 47031,N1(C(C(C)OC)=O)CCCN(C(c2nc(Br)c(C)s2)=O)CCC1 47032,N1(C(CCCC=C)=O)CCC(C)N(C(C2CC(C)(C)CN2C)=O)CC1 47033,C1(C(N(C(C)CNC(C23CC(C2)C3)=O)C)=O)CCCC(C)CC1 47034,c1(C(N2CCC(C)(CNC(CC3CC(OC)C3)=O)C2)=O)ncc(Br)cc1F 47035,n1(C(C)(C)C)cc(CC(=O)NC(C)(CNC(=O)Cc2ccsn2)C2CCC2)cn1 47036,c1(OC)cc(F)cc(C(=O)NCC(O)CNC(C2(C)CC(C)OC(C)C2)=O)c1N 47037,N1(C(c2cc(OC)n[nH]2)=O)CC(NC(C2(CC#N)COC2)=O)CC12CCOC2 47038,CC(C(=O)N1CC(C(C)NC(=O)CSCc2ccccn2)C1)C(C)(C)C 47039,c1(N2CC(C(=C)C)OCC2)cccc(S(=O)(=O)NC2CC23CC(OCC)C3)n1 47040,C(CCCC(CO)NC(c1occ(C)c1C)=O)NC(Cc1c(SC)cccc1)=O 47041,N1(CCN(C(c2cncnc2)C(=O)NC2CCCO2)CC)CCOCC1 47042,Cn1nc2c(cc1=O)CC(NCC1CCCc3cccnc31)CC2 47043,c1(CNC(CCn2cc(C3CCN(C)C3)nn2)=O)ccc2c(n1)OCCO2 47044,C#Cc1ccnc(C(=O)NCC(O)CNC(=O)COCC2CCCCO2)c1 47045,c1(CCC(=O)NC(C)CCCNC(=O)C=CC2CCC2)c(F)cccc1Cl 47046,CC1CN(C(CCc2ccc(Cl)cc2)C(=O)NC2CC2)CCN1CCC(F)(F)F 47047,C1(CNC(N(c2ccc([N+](=O)[O-])cc2)CCC)=O)CC(C)(C)CCC1O 47048,C1(C(=O)NCC(=O)Nc2sccc2CO)CCN(C(=O)C(c2cccnc2)O)C1 47049,CC1CCCC1C(=O)NCCOC1CCN(C(=O)C(c2ccc(Cl)s2)=O)C1 47050,c1(C(N(C)CC2CCCN(C(C(CC#C)O)=O)C2)=O)cc(OC)c(C)c(OC)c1 47051,C1(CN(C(=O)CC2CCOCC2)CC)CCCN(C(=O)CS(N)(=O)=O)C1 47052,C(=O)(C1Cc2c(Cl)cccc21)NCCCNC(C1CC(S(N)(=O)=O)C1)=O 47053,c1(CC)c[nH]nc1C(=O)NCCC1CC(NC(c2cnn(CCN(C)C)c2)=O)C1 47054,C(C)(C)(CC(=O)NCCN(C1CCCCC1)C(c1cc(C)ns1)=O)OC 47055,C1(NC(CC#N)=O)CCN(C(c2cnc3n2CCS3)=O)CC12CCC2 47056,c1(C(N2CC3CN(C(CN(C)CC)=O)CC3C2)=O)cc2c(F)ccc(F)c2[nH]1 47057,N#Cc1cccc(N2CCN(C3CCN(C(=O)COCC4(F)CC4)C3)CC2)c1 47058,CC1(NC(c2cc(C3CCC3)on2)=O)CCN(C(C2CCNC2=O)=O)C1 47059,c1(C(=O)NCC2CN(C(c3c(CC)occ3)=O)CC23CC3)cc2cc[nH]c2cn1 47060,N1(C(C(=O)NCCC2(C)CC2)CC2CCC3CC23)CC2CCCCC12C 47061,C1(NC(C(C)C)=O)CC(CNC(=O)COCCSc2ccccc2)C12CCC2 47062,N1(C(c2cccc(C)n2)=O)CCC2C(NC(c3sccc3CN(C)C)=O)C2CC1 47063,C1(Nc2nccc(C)n2)CC(NC(=O)CCc2ccon2)C12CCOCC2 47064,N1(C(CC=C(C)C)=O)CCC(C2(NC(=O)Cc3nnnn3CC3CC3)CC2)CC1 47065,c1(C(=O)NC2(CC=C)CN(C(C3CC3C)=O)C2)cc(OC)cc(Br)n1 47066,CC(C)CCC(C(=O)NCC1CCSC1)NC(C1CC2(CCCO2)C1)=O 47067,C1(C(=O)NCC=CC(=O)N(CCOC)C)CCCC1C(=O)NC(C)C 47068,c1(C(=O)NCC2CC(C)N(C(c3cccc(CO)c3)=O)C2)ccc(Cl)c(C#N)c1 47069,c1(CC)cscc1C(=O)NCCN(C(=O)CCCc1ccccc1)CCOCCO 47070,c1(N2CCC(NC(C(CC)C)=O)C(F)C2)nc(C)nc(C)c1F 47071,c1(NC(C=CCOC)=O)c(F)cc(F)cc1Br 47072,C1(c2nnnn2C)(N(CC(CC)CC)c2ccccc2)CCCC(C)(C)C1 47073,CCC(CN(C)C)CC(=O)N1CCC1CNC(=O)Cc1nncn1C(C)C 47074,Cn1c(C(=O)NCC2COCC2NC(=O)Cn2ccc(C(F)(F)F)n2)nnc1S 47075,N1(C(C2CCC(C)O2)=O)CC(C)(C)CC1CNC(c1cnc(C2CC2)nc1O)=O 47076,C(=O)(CC1=CCCC1)N1CCC(C(C)C(=O)NCc2cc(C(C)(C)C)n[nH]2)CC1 47077,c1(OCC)ccc(C(N2CCOCC2)CNC(=O)C(C)NC(C)=O)cc1C1CC1 47078,c1(C(=O)NCCC2CC(NC(=O)C(O)C3CC3)C2)cc(F)c(F)cc1F 47079,C(=O)(CN=c1cc[nH]cc1)N1C(C)C(NC(c2c[nH]nc2Br)=O)CCC1 47080,c1(C(=O)NCCOCCCNC(c2n(C)ccn2)=O)cc2c(cc1O)CCCC2 47081,C1(OC)CN(C(c2cc(OC3CC3)no2)=O)CC1NC(=O)CCCOC(C)(C)C 47082,c1(C(=O)NC2CC(CNC(C(COCC)(C)C)=O)C2)ccnc(O)c1Br 47083,CCCCCCCC(O)CC(=O)N1CCNC(C(=O)NC2(CC)CCCCC2)C1 47084,CCC(CC)CC(=O)N1CCC(NC(=O)C(O)CC(N)=O)C1C(C)(C)C 47085,c1(C(=O)NCC(C)(C)OCC(=O)N(CC(COC)C)C)cccc2c1OCO2 47086,C12(CNC(c3c(CSC)cccn3)=O)CCC(CC1)N2C(C1C=CCC1)=O 47087,c1(OC)ccc(F)cc1C1CCCN1CCCCNCCC(C)C(C)C 47088,C1(C)(CC)CC(NC(=O)CC2CCCCC2)CN1C(=O)CC1(OC)CCOCC1 47089,CC(CC(=O)NCC1(C)CCCN1C(=O)Cc1cncn1C)CC(F)(F)F 47090,N1(C(C2(C#C)CN(C(=O)CC(C)(C)OC)C2)=O)CCC2C(CCN2C)C1 47091,CCC(CC(C)C)C(=O)N1CC(CN=c2nc[nH]s2)C(C)(C)C1 47092,C1(NC(C(C)C(C)(F)F)=O)CC2CCC(C1F)N2C(c1ccc2c(c1)CCN2)=O 47093,C(=O)(C1=CC2(CCNC2)C1)N1CCC(C(N(C(C)C)C(C)C)=O)CC1 47094,C12(CNC(C(C)CN(C)C)=O)CC(CCO1)N(C(=O)C(CO)C(F)(F)F)C2 47095,c1(NC)ccc(C(N2CC(CNC(=O)Cn3cccn3)C3(CC3)C2)=O)cc1F 47096,N12CCC(O)(C1)C2=O.N1(CC(=O)Nc2cn(C)nn2)C(=O)CSC1=S 47097,c1(C(N2C(C(C)NC(C3(C)CC(C)C3)=O)CCC2)=O)cn2ccccc2n1 47098,N1(C(CNC(c2n[nH]cc2Cl)=O)=O)CCN(C(=O)C(=Cc2c[nH]cn2)F)CC1 47099,c1(OC)cc(C(N2CCC(C)(NC(=O)CC3CCC3(C)C)C2)=O)ccc1F 47100,OC1CC(CCF)(N(c2ccccc2)C(Cc2ccccc2)C(=O)O)C1 47101,C=CC1(c2cn(CCCF)nn2)COCCN1C(C1CC1(C)C(=O)O)=O 47102,C1(NC(C(C)Cc2ccccn2)=O)CN(C(c2ccc(F)c(I)c2)=O)CC12CC2 47103,c1(C(=O)NC(=O)N=S(C)(C)=O)sccc1C.N(CC)(CC)CC 47104,C1(NC(c2ccc(Cl)nn2)C)CCCN(c2ccccc2)C1 47105,C1(NC(C2CC2(F)F)=O)CCC2CN(C(C3(CO)CC3)=O)CCC2C1 47106,c1(OC)ccc(CC(N2CC(CNC(C3(O)CC3)=O)C(F)(F)C2)=O)cc1Cl 47107,C(CNC(C1CN(C)C(=O)N1)=O)(CC(=O)NC1(CO)CC(C)C1)OC 47108,N1(C(C2CCN(CC)C2)=O)CCC(N(C)C(c2ccn3nccc3n2)=O)C2(CC2)C1 47109,[N-]=[N+]=NCCCCCC(=O)NCC1CCC(NC(c2ccc(C(N)=O)o2)=O)C1 47110,CC1(C)CCC(C(=O)NCC2CN(C(c3ccc(CO)nc3)=O)CCO2)CC1 47111,CCC(C(=O)N1CCC(NC(c2cc([N+](=O)[O-])ccc2O)=O)C1)C(C)(C)CC 47112,C1(O)(CNC(C2(C#C)CCCCC2)=O)CCCN(C(C2(NC(C)=O)CC2)=O)CC1 47113,C(CC1c2ccccc2CCN1C(=O)C(O)C(C)C)NC(C(Br)=C(C)C)=O 47114,C(=O)(CCCC(=O)NC(C)C)N(C(CNC(CSc1nc(C)[nH]n1)=O)C)C 47115,CCC(C)(CCC(C)C)C(=O)NC1COCC1NC(c1cncc2nc[nH]c12)=O 47116,CC(O)CCCCCC(=O)NOCc1cn(-c2ccc3n[nH]cc3c2)nn1 47117,C=C(C)CCCC(=O)N(C1CCN(C(c2ccncc2N)=O)CC1)CCCC 47118,CC(C)(C(=O)N1CCC(Nc2ccccc2)CC1)S(C)(=N)=O 47119,c1(CNCc2cccc(-c3cccc(O)c3F)n2)cnn2c1CCCC2 47120,CC1=C(C(=O)N2CCN(C(c3cscn3)=O)C(CCO)C2)CCS1(=O)=O 47121,S(=O)(=O)(c1cn(C)cn1)NCC(=O)NCC1C(NC(CCc2c(C)noc2Cl)=O)C1 47122,Cc1c(C(=O)NC(C)(C)C(C)NC(=O)C(C)CC(F)F)nn(C)c1N 47123,N1(C(C(CCOC)C)=O)CCC12CN(C(=O)Cc1c(C)cccc1Br)C2 47124,C(CCCCC(=O)N1CCCC1C(C)(C)O)N(C(C(C)CC1CCC1)=O)C 47125,CC1COC2(C1)CN(C(C1CCCN1C(C1CC(CF)C1)=O)=O)C2 47126,N1(C(CC2(NC(c3ccnc(C)c3N)=O)CC2)=O)CC(C)C12CCOCC2 47127,c1(CCC(=O)N(C2CCN(C(c3cc(C)c[nH]3)=O)CC2)CC)cc(F)ccc1F 47128,CC1(C(=O)NC(CNC(C2CCCO2)=O)CO)CCC2CC2C1 47129,C1(C(N(CC(C)NC(c2cccc3nonc23)=O)C)=O)CNc2ccccc2O1 47130,c1(OC)cc(C)sc1C(=O)NC(C1CN(C(=O)CCCC2CCCC(=O)N2)C1)C 47131,C(=O)(CCCCCNC(=O)CC1CC(F)CN1C(c1cc(O)nc(Cl)c1)=O)OC 47132,c1(OC)c(C(=O)NCC(O)CN(C)C(c2cnc(Cl)s2)=O)csc1Cl 47133,c1(SC)c(C(=O)NC2COCC2CNC(C2Cc3cscc3C2)=O)cccc1F 47134,C(=O)(C(C#N)C(C)(C)C)N1CCC(OC)(CNC(=O)CCOCC(F)(F)F)C1 47135,C1(CNC(C2(C(=O)OC)CCCC2)=O)CC2CN(C(c3c[nH]cc3Br)=O)CC12 47136,C(c1ccc(F)cc1F)=CC(=O)NCC1(OC)CCN(C(C2COC(=O)N2)=O)C1 47137,C(=O)(C(O)c1ccco1)NCCCOCCCNC(C1C(CCC)C1)=O 47138,C1(NC(c2ccc(NC)nc2)=O)CCC(C)N(C(=O)CCSC)C1 47139,S(=O)(=O)(c1ccc2nc(C)oc2c1)Nc1c(C)cc(Br)cc1Cl 47140,C(=O)(C(O)C(F)(F)F)N1CCC(C)(CCNC(c2ccc(C#C)o2)=O)C1 47141,C(CN=c1[nH]c(=NCc2cnc(O)[nH]2)c2sccc2[nH]1)C1C(C)C1 47142,C(C(=O)N1CCCc2nccn21)C1(C(CC2C(C)(C)C2)=O)CC1 47143,c1(-n2cc(CCCNC(C3C(C(=O)OC)(C(C)C)C3)=O)nn2)cccc(C)c1Br 47144,C(=O)(CC(CCCC(C)C)NC(=O)CNC(=O)Nc1cc(Cl)cc(Cl)c1)OC 47145,C12CC=CCN1C2=O.C(=O)(C(C)N=[N+]=[N-])NCC(N1CC(OC)C1)=O 47146,C1(NC(c2n(CC)ncc2)=O)CC12CC(NC(=O)C(O)C(C)C)C2 47147,Cc1csc(=NCC(=O)N2CC3C(CNC(=O)CSC4CCCCO4)C3C2)[nH]1 47148,C1(NC(c2ccc(CC)[nH]2)=O)CCN(C(c2cc(C(C)(C)C)oc2C)=O)CC1F 47149,c1(OCCC)ccc(C(N2CC(C)(NC(C3CCCCCC3)=O)C2)=O)cc1 47150,N1(C(CC(=O)OC)=O)CC2CC1C2NC(c1nscc1Br)=O 47151,C1(C(N(C(C)C(=O)NC)CCC)=O)C2CCC1(c1cccnc1)C2 47152,N1(C(Cc2ccn(CC)n2)=O)CC2(CCC(CNC(=O)CCn3cccn3)O2)C1 47153,CS(=O)CCCCNC(C1(CNC(C2CCOC2)=O)CC=CC1)=O 47154,c1(OCc2onc(-c3ccc(OC)cc3)n2)ccc(C(C)=O)c(F)c1Br 47155,C(C1=CCN(C(c2ccnc(N(C)C)c2)=O)CC1)NC(C(CC)NC(N)=O)=O 47156,C(C(C)C(F)C(=O)Nc1cccc(Cl)c1)NC(c1c(OC)nn(C)c1)=O 47157,Cc1ccnc(C(=O)NCC(C2CCCC2)NC(c2conc2C(C)C)=O)c1N 47158,C(CCC(O)C(=O)NC(C)C(O)C(F)F)NC(COCC)=O 47159,C1(C(=O)NCCC(CCNC(c2ccc(C(C)=O)o2)=O)C)CC2(CCCO2)C1 47160,N1(C(COCCN=[N+]=[N-])=O)CCC2(CC1)CC2NC(C1CN2CCC1CC2)=O 47161,Cc1cc(C(N2CC(CCO)(NC(=O)C(C)SC(F)(F)F)C2)=O)cnc1C 47162,C(C(C)CC(=O)N1CCC(CCO)C1)NC(CCc1cnc(C)o1)=O 47163,C1(C(=O)NC2C=CCC2)(NC(C2CCCSC2)=O)CCOCC1 47164,c1(C(=O)NCC2CCC(NC(C3N(CCC)CCC3)=O)C2)c(C)ccc(F)c1N 47165,C1(CC(=O)OC2(CC3CC3)CC2)CCN(CCCF)C1.c1(O)ccccc1 47166,CCCCCCCCC(C)CC(=O)NC1CCC1(C)C 47167,n1(C(C)CC(=O)NC2CCOCC2NC(=O)C2=CSCS2)cnc2ccccc12 47168,C(=O)(C(C)P(C)(C)=O)N1CCC(OC2CN(C(CC(C)OC)=O)C2)CC1 47169,c1(OC)cc(C)c(CNC(C23CC2CN(C(c2cnc(C4CC4)o2)=O)C3)=O)cn1 47170,C1(C(N2CCC(C)(NC(C)=O)C2)C(=O)NCCCOCCO)CC2C=CC1CC2 47171,N(C)(S(=O)(=O)N(C)C)CC(N1C(CN(C(c2ncn(C(C)C)n2)=O)C)CCC1)=O 47172,Cc1cccc(N)c1C(=O)NCC1CCCCN1C(=O)CCNC(=O)CO 47173,c1(N(CCNC(CCC(C)(C)F)=O)CC#N)ncc(Br)cc1C#N 47174,CC(C)CCCC(=O)NCC(CC(=O)Nc1cscc1C1CC1)C1CCC1 47175,C(=O)(CC(O)CC1CCNCC1)N(c1ccccc1)CCOCCC(C)C 47176,Cc1cc(Oc2ccccc2NCc2cccc(C(=O)O)c2)ccn1 47177,N1(CC)CCCN(C(=O)CONC(C2CCOC(NC(=O)NC)C2)=O)CC1 47178,CCC1=NOC(C(=O)NC2(CN(C(=O)C(C3(C4CC4)CC3)C)C)CC2)C1 47179,c1(C(N2CCCC3CNCCC3C2)=O)c[nH]c2ccc(F)cc2c1=O 47180,N1(C(C(C(C)C)=O)=O)CCC(C)N(C(c2cncc(C(N)=O)c2)=O)CC1 47181,Cc1ncc(C(N2CC(C(=O)NC(C)(C)CO)C3(CC3)C2)=O)cc1C#N 47182,C1(CNC(c2c(C)nc(O)[nH]2)=O)CC2CCCCC2N1C(C1CCSC1)=O 47183,C1(C(=O)NC2CCCCN(C(c3ccc(Cl)cc3O)=O)C2)CC2CCCCCC12 47184,C(CC(C)C(=O)NC(C)(CC)CCNC(=O)Cc1nc(C2CC2)cs1)=CC 47185,CC1CCN(C(C2CC(O)C2)=O)CC1CNC(C1(n2cncn2)CC1)=O 47186,C(C1=NOC2CN(C(c3cn[nH]c3)=O)CC12)NC(c1cc(C)c(C)nc1O)=O 47187,c1(C(N2C(C(=O)OC)CC2C)C(=O)Nc2ccccc2)cn2cccc(F)c2n1 47188,N1(C(CC=CCNC(c2csc(Cl)c2)=O)=O)CCCC2(CC2)C1 47189,C1(C)(CNC(c2occ(C)c2)=O)CCN(C(c2ccc(OCCF)cc2)=O)C1 47190,C#CC1(CNC(=O)COCC2(F)CC2)CCCC1 47191,C1(C(=O)NCC2C3CN(C(Cn4nnc(C)n4)=O)CC32)CCN2CCOCC12 47192,c1(CS(Cc2c(C)scn2)(=O)=O)cc(Cl)cnc1F 47193,C(=O)(C(CC1CCOCC1)NC(c1cnn(CC=C)c1)=O)NC(CC=C)C1CC1 47194,CC1CC(C#N)(C(=O)NC2CC(NC(C3(Cl)CC3(F)F)=O)C2)C1 47195,N1(C(C(=O)NCC)=O)CC(C(=O)N(CCCOC)C)C(C2CC2)C1 47196,CCC(C(=O)NCC(C)(C)Cn1cc(-c2cccc(F)c2C)nn1)C(C)O 47197,c1(OCC)ccc(C(=O)NCCCN(CCCNC(c2ncccc2O)=O)C)cn1 47198,N1(C(c2cn(CC=C)nc2)=O)CCC(NC(=O)C(F)C(C)(C)O)CC1C 47199,N1(C(c2nncc(OC)c2)=O)CCC(N(C)C(C2SCCS2)=O)C(C)C1 47200,C1(C(=O)NCC2(F)CC(NC(c3occ4c3CCC4)=O)C2)CCCC2(CCC2)O1 47201,N1(C(C(C)(C)NC(=O)OC)=O)CCC(NC(=O)C(C)(C)C)C(O)C1 47202,C1(CC(=O)NC2CC(CNC(CCCNC(C)=O)=O)C2)COCC(C)(C)O1 47203,N1(C(c2ccc(F)c(C)c2O)=O)CC2(C1)CN(C(=O)CCCF)CC2CO 47204,C(CN=c1[nH]c(=NC)[nH]c(=NCCCCN(CC)CC)[nH]1)NC(C(CCC)C)=O 47205,N1(C(CC2(NC(C)=O)CC2)=O)CCOC(C(C)NC(c2cc(Cl)cnn2)=O)C1 47206,c1(OC)cccc(=NC(=O)Cc2csc(C(=O)Nc3cc(Br)c(C)cc3F)n2)[nH]1 47207,c1(OC)ccc(OC)c(CC(C)C(=O)OCC(COCc2ccccc2)(C)O)c1 47208,C(N=c1[nH]c(N2CC(C)OC(C)C2)nc2ccccc12)c1ccc(C)cc1Br 47209,n1(C(CC)C)ncc2cc(C(=O)NCC3CCN3C(c3ccncc3)=O)cnc12 47210,CC1CCN(C(c2cc(Cl)cs2)=O)C1C(=O)N(C1CC=CC1)C 47211,CCCCCCCC(=O)N1CCCC1CNC(c1c(Br)c(C)nn1C)=O 47212,C1(C(N(CC(O)CNC(C2CC23CCCCC3)=O)C)=O)CCC(=C(F)F)CC1 47213,C1(CC=C)(NC(C2CC2(F)F)=O)CC2CCC(C1)N2C(=O)Cc1c(C)noc1Cl 47214,C1(NC(COCCOC)=O)CCC2(CC1)CCN(C(c1csc3nccn13)=O)C2 47215,C(C(O)C(F)(F)F)C1(CC(=O)OCCNC(C(C)N(C(C)=O)CC)=O)CC1 47216,c1(CCC(=O)NC2CC(C)N(C(=O)CC#N)C2)cc(F)ccc1Br 47217,N1(C(C2CCN(C)C2)=O)CC=CC(C(N2CCN(CC(N)=O)CC2)=O)C1 47218,C1(C(N(CCCF)CC)=O)CC2CC2N1C(C1CC=C(C)CC1)=O 47219,N1(C(CC2(CNC(C3CCN(C)CC3)=O)CC2)=O)CCCC(F)CC1 47220,C(=O)(C1=NOC(C)C1)N1C(C(N(CC(CCC)O)C)=O)C=CC1 47221,N1(C(CCC(=C)C)=O)CCC(C2CC2)(CNC(=O)CC2C(C)(C)C2(C)C)C1 47222,N1(C(c2cnc(C)nc2)=O)CC2CC(C)N(C(C3CCCOC3)=O)C2C1 47223,c1(C(=O)NC(C(C)NC(C2(CC)CC(C)(C)C2)=O)C)ccc(C(F)(F)F)c(F)c1 47224,N1(C(C(=O)NCCCOCCCC)=O)CCCC(NC(C2(CSC)CCC2)=O)C1 47225,c1(CC)cc(C(=O)NCC(C)CNC(=O)CC(CC)C2CCC2)ccn1 47226,Cn1ncc(C(=O)NC2CCCCC2NC(=O)CCc2ncccn2)c1Cl 47227,c1(C(C)C)nnc(SCCCCN2CCOCC2)n1-c1ccc(F)cc1 47228,C1(C(N(C(C)CCNC(=O)C=C2CC2)C)=O)CC(c2ccccc2[N+](=O)[O-])=NO1 47229,C1(CC)CN2CCCC2CN1C(C1=C(C)C(C)=C(Br)SS1)=O 47230,c1(C(=O)NCC2(O)CC(C(=O)NCC(C3CC3)OC)C2)cc(C)oc1C 47231,c12nsc(n1)NC(CC)CNC2=O.C1(C(=O)N(CC)C)CC(n2cnnc2)C1.OC 47232,N1(C(C2CCCCC2)=O)CC(C(N2CCC2CC2CC2)=O)C(F)C1 47233,c1(C(=O)OC)coc(C=CC(=O)NC2CCC(N(C)C(c3snnc3C)=O)C2)c1 47234,C1(CN(C(=O)Cc2n[nH]c(O)n2)C)CCCN1C(C1(CC2CCC2)CC1)=O 47235,C1(NC(CS(CCC)(=O)=O)=O)CCC2CCN(C(c3ccc(O)cc3Cl)=O)C1C2 47236,c1(C(C)OC(C2CC2NC(=O)OC(C)(C)C)=O)ccc(-c2ccccc2)s1 47237,C1(n2cc(CC(C)(C)CO)nn2)CCC(NC(c2cc(F)n[nH]2)=O)CC1 47238,c1(C(N(CCCCNC(c2csc(-c3ccsc3)n2)=O)C)=O)cncc(F)c1 47239,C1(NC(C(Cn2cncn2)NC(Cn2nc(C)oc2=O)=O)=O)CCCC1C1CC1 47240,CCN=c1[nH]cc(C(=O)N(CCC(C)NC(C2CC2[N+](=O)[O-])=O)C)s1 47241,C1(N(C(CCOc2cccc(C)c2)=O)C)CN(C(c2csc(=N)[nH]2)=O)CC12CC2 47242,CC(C)(C#N)CC(=O)NC1CC(NC(C2CCC=CCC2)=O)C(O)C1 47243,c1(N(C)C)cccc(-c2cn(C3CN(C(C4CC=CC(F)C4)=O)CC3O)nn2)c1 47244,C1(N(C2CC2)Cc2cnc(C)n2-c2ccccc2)CC(C)CC(C)C1 47245,c1(OC)ccc(CN2CCC(=CC(=O)NCCOC(=O)C3CC3)CC2)c(F)c1F 47246,C1(CC)(CC)CC(NC(C2CCC3(CC2)CC3)=O)CN1C(c1csc(C)n1)=O 47247,N1(C(C(C)NC(C2CCC2)=O)=O)CCCC(O)(CNC(=O)Cn2nccn2)C1 47248,c1(OC)ccnc(O)c1C(N1CC(NC(=O)Cc2cnsc2)C(C)C1)=O 47249,Cc1cc(C(N2CCN(C(C3CCCO3)=O)CC2)C(=O)NC2COC2)cc(F)c1 47250,C1(S(C)(=O)=O)(C(=O)NC(CNC(C(C)=C2CC2)=O)CC(C)C)CCC1 47251,N(C1CC(C)(C)c2ccccc21)Cc1c(Br)cc(OC)c(OC)c1O 47252,c1(-c2ccc(N3CCCC(NC(CC(C)(C)O)=O)C3)nc2)cc(OC(F)F)ccc1F 47253,C(=O)(C(C(C)(C)O)NC(c1ncncc1N)=O)N1CC(C)SCC1 47254,CCC1=C(C(=O)NCC(F)CNC(=O)CCCOC(C)C)SCCO1 47255,C1(C)(CNC(C(CC)n2cccn2)=O)CN(C(c2cc(=O)n(C)o2)=O)C(C)(C)C1 47256,n1(C2CN(C(CCN(C(CCC)C)C)=O)C2)cc(C2COCC2O)nn1 47257,c1(CNC(C(C2CN(C(Cn3nnc(C)n3)=O)C2)OC)=O)cc(C)oc1C 47258,c1(CCC(N2CC(O)(CCNC(=O)C(C3CCCCC3)F)C2)=O)cncc(F)c1 47259,CCCC(C(=O)N1CC(=O)CC1C(=O)N(C)CCc1cnccn1)OC 47260,c1(C(N2CCCN(C(c3ccccn3)=O)CC2)=O)noc2ncccc12 47261,c1(C(=O)NC(C2CCOC2)CC)cn(CCNC(=O)C(C)SC)nn1 47262,c1(OCC)ccc(C(=O)NC(c2ccccc2)(C)CNC(C2CCCO2)=O)cn1 47263,c1(C(C(C)NC(C2(CO)CCCO2)=O)NC(=O)OC(C)(C)C)ccc(F)cc1F 47264,CN1CCC(O)(CC(N2CCC(NC(=O)CC3C=CCCC3)C(O)C2)=O)CC1 47265,Cc1ccc(CC(N2CCC(C)(C(=O)N(C)Cc3nncn3C)C2)=O)cc1 47266,C12(CNC(CN(CCC)C)=O)CC1CN(C(=O)Cn1ncc(Br)c1C)C2 47267,C1(N(CCOC)C(c2ccon2)=O)CCN(C(c2n[nH]cc2Cl)=O)CC1 47268,C#CC1(C(=O)NCC(CC(C)C)N(C)C)CCN(C(=O)CNC(=O)CN(C)C)C1 47269,Cc1ccc(C(F)F)cc1OCC(N1CCSCC1NC(=O)OCCO)=O 47270,N1(C(C(C)Oc2cccnc2)=O)CCC(F)(F)C(Nc2ncc3c(n2)CCC3)C1 47271,C=C(C)CC(C(=O)NC1CCCCC1N=[N+]=[N-])NC(=O)C(C1CCOCC1)F 47272,c1(OC)noc(C2CC2)c1C(N1CCC(CO)(NC(=O)CC2CC2OC)C1)=O 47273,CN1C(=O)Cc2c(-c3nc(CCCCN(C)C)nn3CCF)cccc21 47274,N1(C(c2c(CC)con2)=O)CCC(CF)(NC(=O)C(C)CSC)C1 47275,C1(O)(CCNC(Cc2n(C)cnc2)=O)CCN(C(c2cnn(CCF)c2)=O)CC1 47276,C12(C(N(C(C3CCCCC3)C)C)=O)CC(CO1)N(C(c1ccc(Cl)cn1)=O)C2 47277,N1(C(c2ccnnc2NCC(=O)NC2CCC2)=O)CCc2ccccc21 47278,N1(CC(=O)N(CCNC(=O)CCc2ncc[nH]2)CC)CCc2sccc2C1 47279,C=C(C)c1cccc(NC(C2CCN2C(=O)C(C(C)(C)C)OC)=O)c1 47280,c1(N(C2CCCN(C(C(c3cccc(C)c3)C)=O)C2)C)ncc(C)c(SC(C)C)n1 47281,c1(-c2ccc(CN3CC(CC)C3)cn2)ccc(OC)c(F)c1F 47282,Cc1c(C(=O)NCC(C)CNC(=O)C2=CCCC2C)c(O)nc2ccccc12 47283,CC1(NC(c2coc(Br)c2)=O)CCN(C(c2ccc(C3(C)CCO3)cc2)=O)C1 47284,N1(C(c2c(C)nco2)=O)CC(C)(CNC(=O)CC2CCCC(=O)N2)CC1(C)C 47285,c1(C(=O)NC2CC(CNC(C3(CC)CC3)=O)C2)cc(Br)co1 47286,C12(C(N3C(C)CC(NC(C(C4CCCCC4)C)=O)C3)=O)CCC(F)(CC1)CC2 47287,CC(C)CC(C)(CNC(=O)Cc1cccc(O)c1)NC(c1ccn(C2CC2)n1)=O 47288,N1(C(C2CCSCC2)C(=O)NC2COC2)C2CCCC1COC2 47289,CC(C)(C)CC(=O)N1CCC(C(=O)NOCC2(C)CC2)CC1 47290,C=C=CCC(=O)NCC1COCC1NC(=O)CCc1cc(OC)no1 47291,c1(N(CCCN(C(c2nc(C)n(C)n2)=O)C)C)nc(Cl)ncc1Cl 47292,Cc1cc(-n2ccnc2)ccc1C(=O)NCCN(C(=O)C(F)C(F)(F)F)C(C)C 47293,C1(OCC)CCCCCC1NC(=O)C(F)Oc1ccc(Cl)c(F)c1 47294,c1(C(N(CC(CNC(c2c(CC)cno2)=O)C)C)=O)ccccc1C1CC1(F)F 47295,Cc1cc(=NCC2(CCCO)CCCC2)[nH]c(NC(c2cccnc2)C)n1 47296,CN1CCC(n2cc(C3CCCN3C(=O)CCn3cnc(C(N)=O)n3)nn2)C1=O 47297,CC(CNc1ncc(COC(C)(C)C)s1)(CO)CO.C1(C=O)(C)CCCC1 47298,C1(C(N(C2CCN(C(c3ncsc3C)=O)C2)CC)=O)CCCC2CC12 47299,N1(C(C2=NNC(=O)C2)=O)CCC2(CC1)CN(C(c1cncc(F)c1)=O)CCC2O 47300,c1(OC)ccc(F)c2[nH]c(C(=O)NCC(C)(CO)NC(=O)CC(C)O)cc12 47301,c1(C(=O)NCC2C(NC(CC3(CC)CCC3)=O)C2)cn(C2CCCC2)nn1 47302,c1(N2CCCC(CCC(C)C)C2)cccc(S(=O)(=O)NCc2csc(Cl)c2)n1 47303,C1(C)(CNC(c2c(CC)con2)=O)CN(C(=O)CC(C(F)(F)F)OC)C(C)(C)C1 47304,C1(NC(c2c(C)cc(SC)o2)=O)CCN(C(c2cn(C)ccc2=O)=O)C1(C)C 47305,C1(C(=O)NCc2nc(C)c(C)o2)CC2(CCN1C(=O)CC1CCC(=O)C1)CC2 47306,c1(CC)cc(C(=O)NC(C2CCN(C(=O)COC(C)C)C2)(C)C)c(C)o1 47307,C1(C)(CC)CCN(C(C2C3CC3CN2C(c2cc(C3CC3)on2)=O)=O)CC1 47308,N1(C(=O)Cc2nc[nH]n2)CCOC2(CCN(C(C3CC4CCC3O4)=O)C2)C1 47309,CC(C)C(CN(C)C)N=c1nc(N2CC3CCC3C2)c2c([nH]1)CCS2 47310,Cc1nc(Cl)[nH]c(=NC2CC(F)(CNC(=O)C(C)CF)C2)c1F 47311,Cn1nc(C(N2C3CCC2CN(C(C2CC24CC4)=O)CC3)=O)c2nc[nH]c(=O)c12 47312,CC(CC(C(=O)c1nn(C)c2c1CCCC2)N(C)C)CC(C)(C)C 47313,C1(C(=O)NCCC(=C)CNC(c2csc(C)n2)=O)CC(=O)N(C2CCCCC2)C1 47314,C1(OC)CN(C(C2CC(C#N)C2)=O)CC1NC(C1(c2ccccc2F)CCC1)=O 47315,c1(CCNC(C2C(C)CNCC2)=O)csc2ccc(Br)cc12 47316,Cc1cnc(NC(C2CC(F)CN2Cc2c(C)cccc2Br)=O)c(Cl)c1 47317,c1(C(N(CCCNC(C(CCCCCC)C)=O)C)=O)cc2n(n1)CC(C)NC2=O 47318,C(C(CC1CC1)C(=O)NC(C)(C)C(C)O)NC(Cc1c(C)occ1)=O 47319,C(=O)(CC(C(F)F)NC(c1n[nH]c(O)n1)=O)NCCC(CC)(C)C 47320,Cc1cc(C(=O)NC2CN(c3ncccn3)C2)n(CC)n1.C1(C(C)N)CCCC(C)C1 47321,C1(C)(C(N2CCC(=CCNC(COCCCCC)=O)CC2)=O)CCC(=O)NC1 47322,CCC(C(C)O)NC(c1ccoc1CNC(=O)COCC(C)C)=O 47323,C1(NC(c2cn3ccsc3n2)=O)CN(C(=O)C(F)(F)C(O)C2CC2)CC1C1CC1 47324,Cc1c(CNC(=O)NCC2(F)CCCCC2)cccc1F 47325,CS(=O)c1cccc(NCc2noc(-c3ccoc3C(F)(F)F)n2)c1 47326,C=CC1(C2(C(=O)NCCCCN(C(=O)CSc3cccs3)C)CCC2)CCC1 47327,C(c1ccc(F)cc1)=C(C)C(=O)N(C)CCN(c1cc(Cl)nc(CS(C)(=O)=O)n1)C 47328,CC1CC(NC(c2cncc(O)c2)=O)CCN1C(c1cccnc1Cl)=O 47329,Cc1[nH]c(C#N)cc1C(N1CC(CC(N2CC3(CCC3)C2)=O)C(C)C1)=O 47330,N1(C(c2c(C)ncnc2)=O)CCC(F)(C(=O)N(CCCC(O)CO)C)CC1 47331,c1(OC(C(N2CCC(C)CC2)C)=O)ccc2ccccc2c1 47332,c1(NC(C2ON=C(C)C2)=O)ccc(NC(=O)CN2C(=O)CCCC2=O)cc1C 47333,C#CCCCC(C)C(=O)N1C(C(=O)NCc2cccc(CC)c2)CC1C 47334,N1(C(c2c(C)csc2Cl)=O)CCC2(CC(NC(c3c(C)ncnc3C)=O)C2)C1 47335,C(CC(O)C(=O)NCCCCC(C)NC(c1ccc(NC=O)cc1)=O)SC 47336,N1(C(c2c(C)nc(C(C)C)cc2)=O)CCC2(NC(=O)CN(C)CCO)CCCC12 47337,Cc1nn(C)c(C)c1S(=O)(=O)NCCC(=O)NCC(C)(C)NC(C1CC1C#N)=O 47338,c1(OC)ccc(CCNC2CC3(NC(=O)OC(C)(C)C)CC2C3)c(O)c1OC 47339,c1(C(=O)NCCCC(C)NC(CC2C(OC)COCC2)=O)nc2cnccc2s1 47340,c1(C(N(C(c2ccccc2)CNC(C2CNC(=O)C2)=O)C)=O)cc2cccnn2n1 47341,C1(SCCNC2CC(c3ccccc3F)(C(=O)OC)C2)CC2CCC1C2 47342,C1(CC(=O)NC2(CC=CC)CCC2)CCCN1C(C1COCCO1)=O 47343,CC(C(=O)NC1C2CCOC2C12CCCC2)N1C(=O)COc2ccccc21 47344,Cn1cnc2c1CCCC2C(=O)NCC1(F)CN(C(=O)CCC2CCOC2)C1 47345,C1(C)(NC(C2(C#C)CCC2)=O)CCN(C(=O)CNC(=O)CNC(C)=O)C1 47346,Cc1cc(C(F)F)nn1CC(N1CC=CC(NC(C2(C)CCOC2)=O)C1)=O 47347,C=Cc1ccc(C(=O)N(C2CCCCN(C(C3(C(C)C)COC3)=O)C2)C)cc1 47348,c1(C(=O)NCC2(O)CCCN(C(CCSC)=O)C2)nc2ccccn2c1F 47349,C1(C(=O)NC(CC)CN(C)C)CCCN(C2CCCCC2OC)CC1 47350,N1(C(C(CCSC)(C)C)=O)CC2CC(C1)CN(C(C1CC3CC(=O)C1C3)=O)C2 47351,C1(OC)CC2(C1)CC2NC(=O)C(C1(O)CCC1)NC(=O)C=Cc1cc[nH]n1 47352,C(CC(O)CC(=O)NC1CCC(N(C(=O)C(C)n2cncn2)C)CC1)SC 47353,N1(C(Cc2c(C)nccc2)=O)CCC(O)(CNC(c2ccc([N+](=O)[O-])o2)=O)CC1 47354,c1(Cn2cc(CSC)nn2)cccc(C(=O)NC(C2CCOCC2)C)c1 47355,N1(Cc2cccc(-n3c(C)cc(C)n3)c2)CCCC(NC(=O)C(C)(C)C)CC1 47356,C1(CC(=O)N(C2(C#C)CC2)C)CC(O)CN1C(=O)CN1CCCC1 47357,c1(C(C)=O)cc(C(=O)NCC23CC(NC(c4cnccc4Cl)=O)(CO2)C3)n(C)c1 47358,N1(C(c2oc(C)c(CO)c2)=O)CC2(NC(C3CC3CF)=O)CCC1CC2 47359,C1(NC(COCC)=O)CC2CC1CN(C(c1cc(C)ccc1NS(C)(=O)=O)=O)C2 47360,C1(C(N2CC(CC)NC(=O)C2)=O)C2CCCC2CN1C(c1cn(C)nn1)=O 47361,C1(NC(=O)C=CCNC(=O)CC2CC=CCC2)CCC(C2CC2)O1 47362,CCC(N)CCC(=O)N1CCC12CN(Cc1ccccc1)C2 47363,C12CCN(CC1O)C2=O.O=C(CC(F)(F)F)NCC(=O)Nc1cnccn1 47364,c1(C(=O)NCCC(CNC(=O)Cc2c(Cl)cnn2C)OC)ccc(F)cn1 47365,C(=O)(C(F)C(F)(F)C(F)(F)F)NCC1CC(NC(C23CCC(OC)C2C3)=O)C1 47366,C1(C(N(C)CCc2ccccn2)=O)CN(C(C2C3CCC(F)C23)=O)CC1(C)C 47367,c1(OCC)ncc(C(=O)NCCC2(NC(=O)C(C)(C)O)CCCC2)s1 47368,N1(C(CNC(C(=O)NC(c2ccc(I)cc2)CC)=O)(C)C)CCC(C)CC1 47369,C1(C(=O)NCCC2CC(NC(C(n3ccc(C(F)(F)F)n3)C)=O)C2)CCCCS1 47370,CC12CC(C(=O)NC3(C4CCCCN4C(c4ccc[nH]4)=O)CC3)(C1)C(C)(C)O2 47371,N1(c2c(Cl)cnc(OC)n2)CCN(C(=O)CCc2cnn(C)n2)CCC1C 47372,C1(NC(N2CC(OCc3c(C)ocn3)C2)=O)CN(Cc2ccccc2)CCN1C 47373,c1(C(=O)NC(CC)CNC(C2COCC(C)(C)O2)=O)ccccc1[N+](=O)[O-] 47374,CCCCC(O)C(C)C(=O)N1CC2CCC(C1)N2C(c1cnn(CC)c1C)=O 47375,O=C(N1CC(n2cc(-c3cnc(C4CC4)s3)nn2)CO1)c1cccnc1C1CC1 47376,c1(CC(=O)NC2CC(C(C(=O)N(C(C(C)C)C)C3CC3)F)C2)cncnc1 47377,c1(C(c2nnnn2C2CCOC2)NC2(CC)CC2)cc(C)ccc1Cl 47378,C=CCCC(C(=O)NOCCF)NC(C1CC=CCO1)=O 47379,C(=O)(CC(C)(C)C(F)(F)F)NCC1N(C(C(C(=O)OC)OC)=O)CC2(CC2)C1 47380,S(=O)(=O)(C(Cl)(Cl)Cl)NC1(C(N(CCC#C)CCC#N)=O)CC1 47381,N1(C(c2c(C)nn(C3CC3)c2)=O)CCC(C)C(NC(=O)Cc2cc[nH]c(=N)c2)C1 47382,N1(C(COCC=C)=O)CC2CC(C(=O)NCCOCCC3CC3)C(C2)C1 47383,CCCCC(C)CCC(=O)NC1CN(C(C23CCC(CC2)CC3)=O)CC1C(F)F 47384,C12(C(N3C(CNC(C4(CCC=C)CCCC4)=O)CCC3)=O)CC(C(F)F)(CO1)C2 47385,N1(C(c2cc(CC)ncn2)=O)CC(C(=O)NCc2cncn2CC)CC(C)C1 47386,C1(OC)CCCN(C(c2cc(CNC(C3CC3C3CCC3)=O)[nH]n2)=O)C1C 47387,C(CNC(=O)CCCc1cnn[nH]1)(CC(=O)N1CCC(N(C)C)C1)OC 47388,C1(NC(c2c(SC)cccc2)=O)CC2CN(C(=O)CCc3cn(C)nn3)CC12 47389,Cc1sc(C)c(S(=O)(=O)NC(=O)CCCc2ncco2)c1C 47390,N1(C(=O)CN(C(C2CC2Cl)=O)C2CC2)CCC(CO)(CO)C1 47391,Cc1cc(-c2nc(CC(F)(F)F)nn2CCCN(C)C)nc2ccccc12 47392,N1(C(C)C)C(=O)CCC1C(=O)OCCC1(C)CC1(F)Cl 47393,C(=O)(C1CCc2c[nH]nc21)N1C(C)C(NC(c2ccc(C(N)=O)nc2)=O)CCC1 47394,C(=O)(C(C(C)(C)C)NC(N)=O)N(CC(F)(F)F)CCN(C)CP(C)(C)=O 47395,c1(-c2scc(C(=O)NC(c3ccc(Cl)cc3)CF)n2)ccc2c(c1)OCO2 47396,C(C)(C(O)C(=O)NCC1CCC(CNC(c2ccncc2C2CC2)=O)CC1)OC 47397,N1(C(c2c(C)nsc2)=O)CC(C2CCCN(C(=O)C(C)(F)F)C2)C1 47398,CCCCC(O)C(=O)N1CC2C(C(=O)NCC(n3cccn3)C)C2C1 47399,C1(C(N2CCN(c3cn(C)nc3)CC2)=O)(C(=O)OC(C)(C)C)CC(O)C1(C)C 47400,c1(C(=O)NCC2(CNC(c3sc(C)c(O)n3)=O)CCC2)c(O)cccc1Cl 47401,c1(NCC(C2CC2)NC(c2ccncc2F)=O)ncc2scc(Br)c2n1 47402,N1(CCCNC(C)CCC(F)F)CC2C3C=CC(CC3)C2C1 47403,N1(C(CC=C(C)C)=O)CCCOC(CCNC(C2(C)CN(S(C)(=O)=O)C2)=O)C1 47404,C1(C(=O)NCC(C)N(C(C2CC(NS(C)(=O)=O)C2)=O)CC)CCCC(=O)N1C 47405,N1(C(C2(CO)CCN(C(CCC3CC(OC)C3)=O)CC2)=O)CC2COCC(C2)C1 47406,O(C1CCCCc2ccccc21)CC(N)CC1CCCC1 47407,c1(CC#N)ccnc(NCC2CCCCN2C(=O)CSc2ccc(F)cc2)n1 47408,S(=O)(=O)(c1ccc([N+](=O)[O-])cc1Cl)NCCCNC(N1CCC(OCC)CC1)=O 47409,C(CCCCCC(=O)N(CCCCCO)C)n1cc(CC)nn1 47410,C1(CC=C)(NC(=O)C(O)C2CCC2)CCCN(C(=O)CCCn2cncn2)C1 47411,C1(C(N(C2CN(C(C3CCC(C)(C)CC3)=O)CC2(C)C)C)=O)COC(C)(C)CO1 47412,C1(NC(C2CC2(F)F)=O)CCCN(Cc2cnn(-c3ccccc3)c2)C1 47413,Cc1cc(C2CC2)cnc1C(=O)N(C)CCNC(=O)CCc1ccccc1O 47414,N1(C(C(CSC)(C)C)=O)CCC2(NC(=O)Cn3ccc(=O)cc3C)CC2C1 47415,N1(C(Cn2ncc(CC)c2)=O)CC(O)CCC1C(=O)NCc1ccc(F)c(F)c1 47416,c1(C(=O)NCC(CCOC)NC(CC(CCC)C)=O)ccc2c(c1)CNC2=O 47417,CC(C)(O)C#CC(=O)NCCCNC(C1(C(=O)NC)CC1)=O.C12=CC=C(C=C1)C2 47418,CC(C)C(C(=O)N(CC(C)CNC(C12CC(CC(F)F)(C1)C2)=O)C)n1cnnc1 47419,C(=O)(CC(O)C(C)C)NC1(COC)CCN(C(=O)CNC(c2ccccn2)=O)C1 47420,N1(C(C(C=C)(C)C)=O)C2CCC1CN(C(c1nc(C3CC3)ncc1Cl)=O)CC2 47421,C1(Cn2cc(C(C)(C)NC(=O)C3CC3)nn2)CN(C(c2ncc[nH]2)=O)CCO1 47422,N1(C(C2CCCO2)=O)CCCC2C1CCCCN2C(=O)COc1cccnc1 47423,N1(C2CN(C(c3cc(COC)sc3)=O)C2)CCN(C(c2ns[nH]c2=O)=O)CC1 47424,C1(C(=O)NC2CC(NC(C3(CC#C)CC3)=O)CC2O)CCc2nnc(O)n2C1 47425,C1(NC(C2C(c3cn(C)nc3)C2)=O)CN(C(=O)CSc2nncn2C)CC1O 47426,C1(C(=O)NC2CC(C(N)=O)C2)CCN(C(=O)CC2CCCC2N(C)C)O1 47427,c1(CC(C(=O)OCC(N2CCC(C(F)(F)F)C2)=O)O)cccc(Br)c1 47428,N1(C(CCCC)=O)CCC2(NC(=O)C(N3CCOCC3)C)CCCCCC12 47429,C(=O)(C(CC(F)F)N(C)C(c1ccc(C#N)cn1)=O)NCC(C1CCCC1)C 47430,N1(C(c2nc(CC)oc2)=O)CCC2(C(=O)NCCn3ccc(C)cc3=O)CC2C1 47431,C#CC1(O)CC(C(N2CCC(N(C(=O)CC(C)(O)C3CC3)CC)CC2)=O)C1 47432,C1(CC)(NC(c2cc[nH]n2)=O)CCN(C(C2CCC(=O)N(CCOC)C2)=O)CC1 47433,C(=O)(CCC(C)C#N)N1CCN(c2nnc(-c3c(C)nc(Cl)s3)n2CCC#N)CC1 47434,Cc1conc1C1CN(C(=O)CC2CC(NC(C3(CO)CCOC3)=O)C2)C1 47435,C#CCCCC(C)C(=O)NC1CN(C(C2(n3cccn3)CC2)=O)CC1C(F)(F)F 47436,C1(C)(CNC(C2CC(C(=O)OC)C2)=O)CCN(C(C2CC2(F)F)=O)C1 47437,C(CCCCC(=O)NC1(C)CC(NC(C2C=C(C)CS2)=O)C1)OC 47438,C1(C(N2CCCC(c3n(CC)cnc3)C2)=O)Cc2c(C)cccc2O1 47439,C12(CNC(C(=Cc3ccco3)C)=O)CCC1CCN2C(=O)CC1=CCCC1 47440,c1(NCC(N2CCC(NC(C3CCCSC3)=O)C(O)C2)=O)ccccc1[N+](=O)[O-] 47441,c1(CC)ncoc1C(=O)NCCCC(=O)NCC(c1ccccc1)F 47442,c1(C(=O)Nc2sc(C(C)=O)c(C)n2)cc(O)ccc1Br 47443,C1(CC(C)=O)(C(=O)OC)CCN(C(CCCC)C(=O)NCCC#C)CC1 47444,C(=O)(CS(=O)(=O)C(C)(C)C)N(CC)CC1CCN(C(c2ccn(C)c2)=O)CC1 47445,C1(CCNC(c2sccc2C2CC2)=O)CCN(C(C2(CF)CC2)=O)C1 47446,C1(NC(C(C)C2CCCO2)=O)CN(C(C2(C(F)(F)F)CCC2)=O)CC(C)(C)C1 47447,N1(C(C2(CC)CC2)=O)CCN(C(CNC(=O)COC2CCCC2)C(F)(F)F)CC1 47448,C(=O)(CCCC(F)(F)F)N1CC(C(C2CC2)NC(=O)C=Cc2ccco2)CC(C)C1 47449,C(CCC(C)C)(C(=O)NCC1CC(C)C1)NC(C1CC=C(C)CC1)=O 47450,C1(C(=O)NCC2(C(C)C)CCCC2)CC2CN(C(=O)C(C)n3ccnn3)CC2C1 47451,C1(CNC(CCC(=O)NC)=O)CCN(C(=O)CCSc2nnnn2C)C12CCC2 47452,c1(-c2n(CC=C)c(N3CCC(=Cc4cccs4)CC3)nn2)n[nH]c2c1CCOC2 47453,c1(OC)cc(C=CC(=O)NCC2CC2NC(C2(n3cnnn3)CCCCC2)=O)sn1 47454,C1(C(=O)NC(COC(C)C)C(=O)NC2CC3CCC(C2)S3)CC12CCCCC2 47455,N(C1CCc2cccnc21)C(CCOCCNC(C1CN2CCC1C2)=O)=O 47456,C1(C(N(C(C)CC(=O)NCc2ccco2)C)=O)CC2CCC2C1 47457,c1(OC)cccc2c(NCc3cccc4c[nH]nc34)ncnc12 47458,C1(C(=O)NC2C(NC(c3n(C)cc(C#N)c3)=O)CCCC2)CCc2nccn2C1 47459,C(=O)(C(C)CC(C)C)N(CCCC(=O)N(CCC)CC)C(C)C 47460,c1(C(=O)NC(CCOC)CNC(=O)C(C)n2ccnc2)ncc(Br)cc1N 47461,c1(C(N(CC(=O)NC2CC(C(C)(C)O)C2)CC#C)=O)nccc2[nH]ccc12 47462,C=CC(C)(O)C(=O)NC(c1ccc(C)cc1)CNC(=O)Cc1csc(C)n1 47463,C(=O)(C(F)(F)C(F)(F)C(F)(F)C(F)F)N1CCCC(NC(C(C=C)O)=O)C1 47464,N1(C(C2(C)CC2(F)Cl)=O)CCC2(CCCC2NC(c2cnc(O)nc2O)=O)CC1 47465,C=C(C)C1OCCCC1C(=O)N(CCNC(=O)C(C)n1cccn1)CC 47466,C(CCC(C)CC(=O)NC1CCCN(C(c2ccns2)=O)CC1)=C(C)C 47467,c1(CC(C)C(=O)N2CCC(N(C(=O)Cn3ccnn3)C)C2)cccc(Cl)c1 47468,CC1CN(C(=O)C(O)C2CC2)CC1NC(c1ncccc1C(F)(F)F)=O 47469,N1(C(C2(NC(CNC(CC)=O)=O)CC(O)C2)=O)CC2(CCC(=O)O2)C1 47470,C#CCCCC(C)C(=O)N1CCC(C)(CNC(c2c(F)ccc(OC)c2F)=O)C1 47471,c1(C(C)C)ccc(C(=O)NCC(C)NC(=O)CCC2CCC(O)CC2)cn1 47472,c1(CN(C)C)ccc(C(=O)NCC2CCCCN2C(C2CC3CCC2O3)=O)cc1 47473,c1(OC)ccc(C(N2CC(OCCNC(=O)C(N)=O)C2)=O)c2ccoc12 47474,N1(C(CSCC(C)C)=O)CC(CNC(=O)CN2CCN(C3CC3)C2=O)CCC1C 47475,C12(NC(CCc3nnc(C)n3C)=O)CCN(C(=O)CC3CCC3)CC1C2 47476,Cc1c(C(=O)NCC(C(C)(C)C)NC(=O)C(C)OC(C)(C)C)nn2ccccc12 47477,C(=O)(Nn1cccn1)C1N(C(c2ccccc2F)CCc2cc(=N)[nH][nH]2)CCC1 47478,C(=O)(C(C#N)C(C)(C)C)NCC1(F)CCC(NC(COCCOC)=O)C1 47479,c1(NC(C2N(C(c3ccc(Cl)cc3)=O)CCC(=C)C2)=O)cnc2c(c1)CCC2 47480,Cc1ccc2c(C(N3CCCC(NC(=O)CC(O)C(C)(C)C)CC3)=O)c[nH]c2c1 47481,c1(CN2CCC(c3cccc(C)c3)C2)c(Br)cncc1Br.C12CCC(C1)NC2=O 47482,N1(C(CSCC=C)=O)CCCCC12CC(NC(c1ncsc1CC)=O)C2 47483,N1(C(C2(CC#C)CCOC2)=O)CCC(CC=C)(NC(c2ccc(CO)nc2)=O)C1 47484,C1(C(N)=O)CC(C(=O)NCCCNC(=O)CSCC2CC2)=NO1 47485,N1(c2n(C)c(C3(O)CCSC3)nn2)CCC2(CCCCO2)C1 47486,N1(C(CC(=C=C)C)=O)CC(NC(=O)C(C)SC)C(N=[N+]=[N-])C1 47487,C1(C(=O)NC2(C)CC(NC(C3CCC(C)CC3)=O)C2)CCn2c(O)nnc2C1 47488,Cn1nccc1CCC(=O)NC1CCCC1NC(c1coc(Cl)n1)=O 47489,Cc1cc(=O)cc(CNC(C2CN(C(c3sccc3C#N)=O)CCO2)=O)[nH]1 47490,C1(NC(C(CC)C#N)=O)CC(O)(C2CCN(C(c3csc(C)n3)=O)CC2)C1 47491,N1(C(=O)Nc2cc(C(=O)OCC)n[nH]2)CC2CC2(CC)C1 47492,n1(CC(=O)Nc2c(F)cc(I)cc2F)ccc(=NC(=O)c2cc[nH]c2)nc1O 47493,c1(C(N2CCC(NC(c3cc(CO)ccc3O)=O)CC2)=O)cn2c(n1)CCC2 47494,C1(CNC(C23NCC(COC)(C2)C3)=O)CCCC2CCCCC12 47495,N1(C(C(CC#C)(C)C)=O)C2CCC1C1CC1(NC(C1CCC(=O)N1CCC)=O)C2 47496,c1(C(C(=O)NC23CN(C(C(C)O)=O)C(C2)C3)=O)cc(F)ccc1F 47497,c1(C(=O)NCC(CN(C(Cc2ccc(C)s2)=O)C)O)nc[nH]c2nccc1-2 47498,C1(C(=O)NC(Cc2ccco2)CO)(NC(Cc2c(C)ccs2)=O)CCCCC1 47499,C1(NC(=O)C=CC=Cc2cccs2)CCC12CN(C(=O)C1=NNC(C(F)(F)F)C1)C2 47500,N1(C(CC(=O)OCC)=O)CC2(CCCC2)C1C(=O)NC(c1nccn1C)C 47501,C1(c2cn(CC(=O)NCC)nn2)CCCCN1C(C1CC1C1CCCO1)=O 47502,S(=O)(=O)(c1cc(C)cnc1NC(CCO)c1ccco1)NC(CCCC(=C)C)C 47503,C(=O)(CN=c1cc[nH]cc1)NCC(C(=O)NCC(CCC)C)C 47504,C1(NC(C2C(=C)CC2)=O)CN(C(c2cc(Br)cn2C(C)C)=O)CC1F 47505,C(C)(C)(CC(=O)NCCC(N1CCC(O)(C(C)C)C1)=O)OC 47506,C1(C(=O)NC(C)CN2CCN(C(c3ccon3)=O)CC2)CC12CCCCC2 47507,c1(CC)cc(NC(C2CCCCC2NC(=O)CCc2ccncc2)=O)cnc1C 47508,c1(C(N2CCC(F)(C(=O)NCC3C(C(C)C)C3)C2)=O)cnn(C)c1C#N 47509,c1(C(=O)NC(CNC(c2cnc(CC)s2)=O)C(C)C)cnn2ccnc(N)c12 47510,N1(C(c2ccc(C(C)(F)F)nc2)=O)CC2=C(C1)CN(C(=O)Cc1cc[nH]c1)C2 47511,C1(CNCc2cnc(C#N)c(F)c2)CC2(CCC(F)(F)CC2)CO1 47512,C(=O)(C#CC1(CC)COC1)N1CC2CCC(N(C(C3(SCC)CC3)=O)C)C2C1 47513,c1(C(=O)NC2(C3CN(C(C(C)(C)CC4CC4)=O)C3)CC2)c[nH]c2ccc(F)cc12 47514,C#CCCCC(=O)NCCN(C(=O)C=CCCC(CC)=C(C)C)CCOC 47515,C1(NC(C2CCCOC2)=O)CC2(C1)CC(C(=O)NCC(O)C(F)F)C2 47516,CC1(F)CN(C(c2ccoc2CC(N)=O)=O)CCN(C(=O)CCS(C)(=O)=O)C1 47517,C(=O)(C1CCCn2ccnc21)NCCC1N(C(c2ncn(CC)n2)=O)CCSC1 47518,c1(CCC(=O)NC2CC(NC(C(C)CSC(F)(F)F)=O)C2)ccc(O)nn1 47519,Cc1ccc(N)c(C(N2CC(NC(=O)C(C)CSC(F)(F)F)CC2CO)=O)c1 47520,C(=O)(C(C)(C)C1=CCN(C(=O)CCCCC(C)CC)C1)N1CC(C#C)(F)C1 47521,c1(Cc2onc(C(=O)NCC)n2)cccc(Br)c1O 47522,C1(CNC(C=CC=CC)=O)CN(C)CCN1C(C1CCCN1CC(C)C)=O 47523,N1(C(C2(c3ccccc3F)CC2)=O)CCc2c(C(=O)O)cccc2C1 47524,c1(CC(=O)N(C2CN(C(=O)C(O)C3CC3)C2)C)ccc(S(N)(=O)=O)s1 47525,c1(CNC(C(C2CCN(C(C(OC)OC)=O)C2)C)=O)cnn(C)c1O 47526,CCC(F)(C(=O)OC)C(=O)N1CCOC(CN(C(=O)Cc2cnoc2)C)C1 47527,CC(N=[N+]=[N-])C(=O)N1CCCC1CN(C(=O)C=CCN1CCCC1)C 47528,S(=O)(=O)(CCCCCl)N1CC(NC(c2occc2Br)=O)C(F)C1 47529,c1(SC)cn(C)nc1C(=O)NC1CCCCC1NC(=O)C(C)NS(C)(=O)=O 47530,N1(C(c2c(C)ccnn2)=O)CC(NC(c2ncccc2Cl)=O)CC12CCOC2 47531,C1(NC(CCC(N)=O)=O)CCN(C(C2CN(C3COC3)C2)=O)C(C2CC2)C1 47532,c1(C(=O)NCCC2CCN(C(C(C)CCO)=O)C2)c(O)cnc2ccccc12 47533,CC(C)(O)C(F)(F)C(=O)NCC1(O)CC(NC(C23CCCC2(C(N)=O)C3)=O)C1 47534,N1(C(C(C)CSC(F)(F)F)=O)CCC(CF)(NC(=O)C(=O)NCCC(N)=O)C1 47535,c12ccc(o1)CCC(=O)N2.C(=O)(CNC(=O)C=CC(=O)N(C)C)N(C)CC 47536,N1(C(CC2(OC)CCC2)=O)C(C(=O)NCC(=O)OC(C)C)CCC1C1CCCC1 47537,C(=O)(CC(=O)NCc1n[nH]cc1C(N1CCCC1CCCO)=O)N(C)C 47538,C(=O)(C(C(F)(F)F)C(F)(F)F)NCCC1N(C(c2ncn(CC)c2)=O)CCOC1 47539,Cc1cc([N+](=O)[O-])ccc1C(=O)NC1CCC1NC(=O)C(=O)NC(C)C 47540,Cc1ccc(C(=O)NC2CCC2CNC(C2COCCO2)=O)cc1Cl 47541,C1(C)(C(N2CC(C(C(N3CCC4CCC34)=O)OC)C2)=O)CC(=O)N(C)C1 47542,C1(C(N(CC(C)NC(C=CC)=O)C)=O)CCCN1CC(C)C 47543,N1(C(C(COC(C)=O)C)=O)CCCC(CNC(c2nc(Cl)c(Cl)s2)=O)C1 47544,C1(c2ccc(C)o2)CCCCCN1C(=O)Cc1ccccc1C(N)=O 47545,C1(NC(C2(OC)CCOCC2)=O)CN(C(C2COCCOC2)=O)C(C)(C)C1 47546,CC1CCCC=C1C(=O)N1CCCN(C(C2CNC(=O)CC2(C)C)=O)CCC1 47547,C(C)(C(C)(C)NC(c1cccn1C1CCCC1)=O)NC(C(C)n1cncn1)=O 47548,c1(CCCC(=O)NC2C(NC(C(CCC)NC(N)=O)=O)C2)cc(O)ccc1C 47549,CCC(C(=O)N1CCC(NC(=O)CCOCc2ccccc2)C1C1CC1)C(C)C 47550,N1(C(c2scc(C)c2)=O)CCC2(NC(c3nc(Cl)ccc3N)=O)CC2C1 47551,C(C(C)(C(=O)NCc1cccc(Cl)c1)NC(c1ccc(F)cc1)=O)SC 47552,C1(N(C(CCOCC#C)=O)C)CN(C(=O)CCCCC)CCC1O 47553,CC(C)(O)CCC(=O)NCCC(F)Cn1cc(CN2CCNC(=O)C2)nn1 47554,c1(C(=O)NCCC2CN(C(C3C(C)C3C)=O)C2)n[nH]c(C2CC2)c1Cl 47555,C(CCN(C)C(C12CC(C)(CO1)C2)=O)(C(C)(C)C)NC(CCC=C)=O 47556,c1(C(=O)NCC2OCCC(NC(=O)CCF)C2)ccc2c(c1)C(=O)CCCC2 47557,c1(NC(CN(C(C2CC2(Cl)CC)=O)C)=O)cn(CCF)nc1C 47558,C1(C(=O)NC(C#C)CC2CC2)CCCCCC1NC(C1(C)CNC(=O)N1)=O 47559,C(=O)(CCCCCCCC(=O)NCCNCc1ccc2cn(C)nc2c1)OC 47560,C(CN=c1[nH]c(=NC2CC2)[nH]c2ccsc12)N(S(=O)(=O)c1cccs1)C 47561,C1(NC(c2nc(C)n(C)c2)=O)CC12CCN(C(=O)C=CC1CCCC1)C2 47562,C(C1=NOC2CN(C(c3ocnc3C(F)(F)F)=O)CC12)NC(CCCC(=C)C)=O 47563,C(=O)(CC(C)(O)C1CC1)N(C1CN(C(c2cscn2)=O)C1)C 47564,Cc1[nH]c(C(=O)Nc2nn[nH]n2)c(C)c1C(=O)Nc1nc(Cl)ccc1O 47565,N1(C(c2cc(C)[nH]c2C)=O)CCCC(C)(NC(c2cnoc2C)=O)C1 47566,c1(C(=O)NCC(C)(C(C)C)NC(C=CCC)=O)c(Br)ccc(C)c1F 47567,N1(C(c2c(NC)cccc2)=O)CCCCC(NC(C23CC(C)(CO2)C3)=O)C1 47568,c1(-c2n(CCOC)nc(CCC(C)C)n2)c[nH]c2ccc(Cl)cc2c1=O 47569,n1(CC(CNC(C2CC(n3ccnc3C3CC3)C2)C)C)cc(C2(C3CC3)CC2)nn1 47570,C1(C(N(CCCNC(C=CCCC)=O)CC2CCCC2)=O)CC12CCCCCC2 47571,c1(NC(N(C)CC2CCC(c3nn[nH]n3)C2)=O)cncc(C(=O)NC2CC2)n1 47572,N1(C(C2(C(N(C)C)=O)CC2)=O)CCn2ncc(CN(C)C(C3CCSC3)=O)c2C1 47573,Cc1cnc(NC(=O)CC2CC(NC(c3cnc(O)c(Cl)c3)=O)C2)c(Cl)c1 47574,C(=O)(CC1=CCOCC1)NCC1CCC(C(N2C(CC)CCC2)=O)CC1 47575,CCC(C)C(O)CC(=O)N1CC2(C1)CN(C(c1c[nH]nc1Br)=O)C2 47576,Cc1ccn2cnc(C(N3CC4CC3CN(C(c3cccnc3S)=O)C4)=O)c2c1 47577,n1(CC)cc(Cl)c(C(N2CCC(O)(CN(C)C(C3(C)CSC3)=O)C2)=O)n1 47578,c1(C(=O)NCC2(NC(=O)CC3CCC(O)C3)CCOCC2)cnc2[nH]nnc2c1 47579,c1(C(=O)NCC=CCNC(C(CC)(C)C#N)=O)nc2ccc(Br)cn2c1F 47580,C1(C(C)C)(C(=O)Nc2cnsc2)CCN(C(c2ccncc2O)=O)C1 47581,C12(C(=O)NC(C3CCCNCC3)C)CCCCC(=O)N1CCC2 47582,c1(C(N2C(C(=O)Nc3cnccc3I)CC(C)C2)=O)ccc(Cl)c(C(F)(F)F)c1 47583,CCCC(C(=O)N1CC2CC1C2CNC(c1cc(C)n(C)n1)=O)OC 47584,C1(C(=O)NC(CCCNC(C(CC=CC)CC)=O)(C)C)OCCOC12CCC2 47585,N1(c2cc(C)nc(N3CCC(C4CCCO4)C3)n2)CCC2(CCOC2)CC1 47586,C1(CNC(C2(NC(c3nc(C)sc3C)=O)CSC2)=O)CCCN(C)C1=O 47587,c1(C(N(C2CN(C(=O)COCCCF)CC2F)C)=O)cccc(Cl)c1F 47588,c1(OC)cncc(C(N2CC(CNC(=O)CC3(C#N)CC3)CC2C)=O)n1 47589,C1(N(C(CC=CC)=O)CC(C)C)CCN(C(C2CCCCN2C(=O)NC)=O)CC1 47590,c1(C(N(C2CN(C(C3CN(C4(CC)CC4)C(=O)N3)=O)C2)C)=O)ccc(=N)[nH]c1Cl 47591,C1(NC(C=CC(N)=O)=O)CCCC2CN(C(=O)Cc3nc4c([nH]3)CCCC4)CC12 47592,N1(C(CCCC#C)=O)CCC2(NC(c3n[nH]cc3OC)=O)CCCCCC12 47593,c1(C(N(CC(CC)NC(c2cccn2Cc2ccncc2)=O)C)=O)cc(C)sn1 47594,c1(C(N(C)CCOCCNC(C2CCCN2S(C)(=O)=O)=O)=O)cc(Cl)n(C)n1 47595,c1(CC)ncc(NC(=O)NC2CCN(CC3CCOCC3)CC2)c(C)n1 47596,c1(C(N2CC(CNC(CC(C)(C)C)=O)OCC2)=O)cc(Cl)ncc1O 47597,C1(CC)CN(C(c2scc(C)c2Cl)=O)CCC1NC(=O)CCc1cccnc1Cl 47598,Cc1cnc(CN(C)C(C2C3CN(C(=O)CCCC4CC4C)CC23)=O)cn1 47599,c1(C(N(C)CCNC(C2CC(CF)C2)=O)=O)c[nH]cc1-c1ccccc1 47600,N1(C(C2C(C)=CCS2)=O)CCC(NC(C2CS(=O)(=O)C2)=O)C(C)(C)C1 47601,CC1(C)CC(NC(=O)CC2(C3CC3)CC2)CN1C(=O)CC1CN2CCC1CC2 47602,C1(C2CCN(C(=O)CC3CCNC3=O)C2)(NC(c2nnc(O)nc2O)=O)CC1 47603,N1(C(C(C(C)C)C2CCC2)=O)CC(NC(=O)CC2CC3(CC3)C2)C2(CC2)C1 47604,C(C)(c1cccc(Cl)c1)=CC(=O)NC(CC)CN(C)C(c1cccc(C)c1F)=O 47605,C12(CCNC(=O)NCc3cn(CCC)nc3)CCC(CC1)CC2 47606,CON1CCC(NC(C2(NC(=O)CC3CC4CC4C3)CC(F)C2)=O)CC1 47607,C(=O)(C(C)(C)C(=O)NC(C)C(C)NC(=O)CNC(c1ccccn1)=O)NC 47608,c1(COCC(N2CC(C)S(=O)CC2)=O)nc2ccccc2s1 47609,N1(CC(=O)N(C(=O)C#CC(C)C)CC)CCc2nnc(Cl)cc2C1 47610,C1(C(N(C(C2CCOCC2)C)C)=O)CCCC(NC(=O)Cc2cccnc2O)C1 47611,C1(CC(=O)N(C(C)CN(C(=O)CN2CCCC2=O)C)C)CC=CCN1C 47612,N1(C(C(C)Oc2cccc(Cl)c2)=O)CC2CCN(C(C3CC=CC3)=O)CCC2C1 47613,c1(CC)cccc(NC(=O)CCOCCNC(C2CC3(CC3)CO2)=O)c1 47614,c1(C(=O)NCC(CO)NC(c2sccc2Cl)=O)ccc(Br)cc1Cl 47615,N1(C(C(=O)NC(c2cccc(OC)c2)CF)=O)CC2CC(C)C2C1 47616,c1(C(=O)NCC2CCCN(C(CCC=C)=O)CC2)nnc2n1CCCCC2 47617,C1(OC)(CNC(=O)Cc2ccc(F)cc2F)CCN(C(=O)CSC(=N)N)CC1 47618,CC(CN(C)C)CCC(=O)N(CCCN(C(=O)C(c1ccc(F)cc1F)=O)C)C 47619,C(=O)(CC(C(C)(C)C)NC(c1c[nH]c(=NC)s1)=O)NC(CCC)C(F)(F)F 47620,N1(C(C(CC)(C)C#N)=O)CCC=C(C(=O)NOCCOc2ccccc2)C1 47621,CC#CCC(C(=O)NC1CCN(C(C)C)C1=O)NC(=O)CCC(C)(C)OC 47622,n1(CC)ccc(C(N2CC(NC(=O)Cn3ccnn3)CC2C)=O)cc1=O 47623,N1(C(C2OCCN(C)C2)=O)CCN(C(c2cnn(C)c2Cl)=O)CC(CO)C1 47624,N1(C(COCC(C)C)=O)CC2CC1CCC2NC(=O)CSCc1cscn1 47625,CN1CC=C(CCNC(=O)C(C)(CO)NC(=O)Cc2ccccc2O)CC1 47626,c1(N2CCC(NC(CC(CCC)N)=O)C2=O)ccc2c(c1)OCCO2 47627,C1(C)(CC(=O)NC(CC2CN(C(CNC(C)=O)=O)C2)C)CCCO1 47628,C1(O)(C(=O)NC(CNC(c2n(C)nc(C)c2Cl)=O)C)CCCC(C)(C)CC1 47629,N1(C(CN(CCC)C(c2cc(COC)on2)=O)=O)CCCC2(CC2)C1 47630,CC1=NN(C)C(=O)C1CC(=O)NC1CC(NC(C2CC(F)(F)C2(C)C)=O)C(O)C1 47631,C1(CNC(Cc2c(C)ncs2)=O)CCCN(C(C2CCC(C(C)C)CC2)=O)C1 47632,c1(C(N2CC(C)(CCC(=O)NC3C(C)CC3)C2)=O)ccc(N)cn1 47633,c1(C2(C(=O)NCC3CCN(Cc4nc(Br)cs4)CC3)CCCC2)ccc(Cl)cc1 47634,C1(C(N2C(CNC(C(c3ccccc3)NC(CC)=O)=O)CC2)=O)(SC)CC=CC1 47635,C1(C(=O)NCC(CCNC(C(N2CCOCC2)C)=O)O)CCCC(F)(F)C1 47636,C1(C)(C(N2C3C(NC(CC4(OC)CCC4)=O)C(C3)C2)=O)CCC2(CC1)OCCO2 47637,c1(C(=O)NC2CCN(CCCCc3ccccc3)C2)ccc2cc(Br)ccc2c1 47638,CC1(CNC(c2cccc(O)n2)=O)CCCN1C(=O)CCc1cnc[nH]1 47639,S(=O)(=O)(c1cccnc1NCC1(CC#N)CC1)NCC(CCOC)(C)C 47640,C1(C(N2C(CN(C(=O)CSc3nncn3C)C)CCC2)=O)CC2C=CCC(C1)C2 47641,c1(C(c2cn(CC(=O)NC(C(C)C)c3nc[nH]n3)nn2)O)cccc(C(=O)O)c1 47642,c1(C(C)(C)C)ccc(C(=O)NC2CCC(CNC(=O)Cn3cnc(=N)[nH]3)C2)nc1 47643,C(=O)(C1CC(=O)Nc2ncccc21)NCC(C)(C)NC(c1cnc(C2CC2)s1)=O 47644,C(=O)(C(C)(C)CCCNC(c1coc(C(N)=O)c1)=O)NC1C(O)CCC(C)C1 47645,C(=O)(C1CCc2c[nH]nc21)NC1CC2CC(NC(CCNC(=O)NC)=O)C2C1 47646,C1(CNC(c2nccc(C)c2)=O)CN(C(=O)C(F)=C2CCC2)CC(C)(C)C1 47647,c1(NC(CC)=O)cncc(C(N2CC(NC(c3cccnn3)=O)C(C)C2)=O)c1 47648,N1(C(CCC)=O)CCCC1CNC(C1CC(NC(=O)C(C)(C)NC(C)=O)C1)=O 47649,C1(C(=O)NC2CC(C)N(C)C2)CN(Cc2cn(C(C)(C)C)nn2)CCC1O 47650,C1(NC(c2cncc(CO)c2)=O)CC12CC(NC(c1cc(C3CC3)ccn1)=O)C2 47651,c1(C(=O)NCC2C3N(C(C(C)O)=O)CC(CC3)C2)ncnc2c1ncn2C1CC1 47652,c1(C(=O)NCC(C)(C2CC2)NC(CN(CC)CC)=O)cccc(CS(C)=O)c1 47653,N1(C(c2c(O)ccc(C)c2)=O)CC2(NC(C3CCCCS3)=O)CCC1CC2 47654,C(=O)(CC(O)CN(C)C)NCC(C)(C1CC1)NC(c1cc(C)[nH]n1)=O 47655,N1(C(c2cc(C)no2)=O)CC2CCCC(NC(=O)C(C)CC3CCC3)(C2)C1 47656,C1(CC(=O)N(CC#C)CC)CCCN(C(c2ccc(SC)o2)=O)C1 47657,C(=O)(CS(=O)(=O)C1CC1)NCC(C1CCN(C(COCC=C)=O)CC1)O 47658,O=C1OCCC12CCN(Cc1nnc(C(F)(F)F)o1)CC2 47659,CC1(C(=O)NC2CCOC2)CCCN1C(=O)CCC1CCOCC1 47660,N1(C(C(CCC)F)=O)CCN(C(=O)CC2COC(=O)C2)CC1CCC 47661,C1(CNC(C(CC2CCC2)OC)=O)CN(C)CCN1C(=O)CC1CC1 47662,C(c1cccc(Cl)c1Cl)=CC(=O)NCCCCCCNC(=O)CC1CCOC1 47663,CONC(=O)C(=O)NCC(C1CC1)NC(c1nnc(S)n1C)=O 47664,C1(c2nn[nH]n2)(C(N2C(C(N(CC(N)=O)CC3CC3)=O)CSC2)=O)CCOCC1 47665,N(C(=NCCCCN1CCN(C)CC1)NC1CC1C)CCOCC(=O)OC 47666,c1(C(=O)NC(CC)CCC(=O)NCC(N2CCOCC2)=O)ccc2c[nH]nc2c1 47667,C(C(=O)OC(C)(C)C)=CCC.C(C(C1CC1)N(C(=O)CN(C=O)C1CC1)C)OCI 47668,CCC(CC(=O)NCC(C)(O)C1CCCC1)NC(=O)C(C)OCCOC 47669,C(=O)(C(CCOC(C)(C)C)N(C)C)NC(C1CCN(C2CCCCC2)C1)C 47670,c1(OC)cc(C(N2CCC(O)(C(C)NC(=O)C=Cc3ccco3)C2)=O)ncn1 47671,C(CC(CC)C(=O)NCC1CCC12CN(C(c1csc(SC)n1)=O)C2)=CC 47672,c1(C(=O)NC(C)CCNC(=O)CSC(F)(F)F)cnn(CC(F)(F)F)c1 47673,c1(C(=O)OC2CN(CCC)C(=O)C2)c(C)nn2c1CN(C(=O)OC(C)(C)C)CC2 47674,c1(SC(c2nc(C[Si](CC)(C)C)on2)c2ccccc2)cnc(O)cc1O 47675,n1(CCCC)nc(C(=O)N(C)CC2(CO)CC2)ccc1=O.C1(=O)C(OC)N1 47676,c1(CC)c(C(N2CC(c3ccccc3C(=O)O)(O)C2)=O)cnn1C1CCCC1 47677,C1(CNC(C2CCC(C#C)CC2)=O)CC2(CCC2)CN1C(=O)CCCSC 47678,N1(C(c2c(C)snn2)=O)CCCC(C(=O)OC(C)(C)C)C1.C12CC(C1)CNC(=O)C2 47679,C1(n2cc(CNC(=O)OCC)nn2)CC2CCC1(NC(C1(F)CCOC1)=O)C2 47680,C1(F)(C(=O)NC2CCC(C(=O)NC(C)Cc3ccccn3)C2)CCOCC1 47681,Cc1nccnc1C(=O)NCCC(C)(C)NC(C1CC(F)(CF)C1)=O 47682,c1(C(N2CCC(NC(C3C(CC)C3)=O)C2)=O)cccc(OC)c1Cl 47683,c1(CC(C)C)ccc(C(C)C(=O)N(CCCN(C)C(c2csc(Cl)n2)=O)C)cc1 47684,C12(NC(c3cc(C4CC4)[nH]n3)=O)CCCC(CN(C(=O)C(F)F)C1)C2 47685,N1(C(c2c(OC)cncn2)=O)CCC(F)(F)C(CNC(c2cc(Cl)c[nH]2)=O)C1 47686,S(=O)(=O)(c1ccc(F)cc1)Nc1ccc(SCC(N2CCOCC(O)C2)=O)cc1 47687,c1(OC)cc(F)c(C(=O)Nc2cccc(NC(C3CC4(CCC4)C3)=O)c2)cc1F 47688,C#Cc1cccc(C(=O)NCC2(OC)CN(C(C3CCC(C)CC3)=O)C2)c1 47689,N1(C(CCc2cccc(OC)c2)=O)CCC2CN(C(C3CCCS3)=O)CC12 47690,C1(CCC(c2nnnn2CC2CCCCC2)NC(C)C2CC2)CC(F)(F)C1 47691,c1(NCC(=O)NCC=CCNC(c2c(C)ccnc2)=O)ccc2ccccc2c1 47692,CC1(C)CC(CC(N2CC(O)CC2CNC(C2CC=CCC2)=O)=O)CC(C)(C)O1 47693,c1(CC)ccsc1C(=O)N(CC(C)C(=O)N(CC(CC)OC)C)C 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47712,CC1CC(S(C)(=O)=O)CN1C(=O)C(=O)NC1CC2CC1CO2 47713,C1(C2CCC2)(C(=O)NCC(C)(C)OCCNC(C2CCC(F)(F)C2)=O)CCC1 47714,C=CCCCCCCC(=O)N1CC(CC(=O)NCC2(O)CCC2(C)C)C2(CC2)C1 47715,c1(C(=O)NCC=CCNC(=O)CC23CCCC2C3)cc2cccnc2o1 47716,C1(NC(C2(CC)CCNC2=O)=O)CC=C(C(=O)N2CC(C(=O)OC)C2)C1 47717,CC1CCc2ncc(C(N3CCCC34CCN(C(c3ccccc3)=O)C4)=O)n2C1 47718,C1(NC(c2ccnc(C)n2)=O)COC2(CCN(C(c3cnsn3)=O)C2)C1 47719,Cn1cc(Cl)cc1C(=O)NCc1ccoc1C(=O)NC1CCCC(F)C1 47720,N1(C(CC=C)=O)CCC2CN(Cc3ccc(Br)cc3O)CC12 47721,CCC(CC)(CCNC(=O)C(=O)C(C)(C)C)NC(=O)COC(F)F 47722,N1(C(C23OCC(C)(C2)C3)=O)CCCC2(NC(c3csc(C4CC4)n3)=O)CC2C1 47723,c1(NC)ncccc1C(=O)NCCC(O)CNC(=O)CCC1CC(C)C1 47724,c1(C(=O)NC2CC(NC(C=CCOC)=O)C2)cc2c(nc1O)CCCC2O 47725,C1(NC(C(CSC)C)=O)CCC2(CCN(C(c3ccoc3Cl)=O)C2)C1 47726,C(CCC(c1ccccc1)NC(N)=O)NC(C(C)O)=O.C(COCCOCCO)SC 47727,Cc1nc(NC(C2CN(C(c3cccc(O)n3)=O)CCC2(F)F)=O)c(F)c(Cl)n1 47728,c1(OC)ccc(C(=O)NCC2(CC(C3CC(=C4CC4)C3)=O)CCC2)c(Cl)n1 47729,CCCCCC(O)C(=O)N1CC2=C(C1)CN(C(c1ncc(Br)cc1N)=O)C2 47730,c1(C(=O)NCC(C)N(c2ncc(C)c(O)n2)C)ccc2nnc(O)n2c1 47731,C#Cc1nccnc1NC(C1CC1NC(c1cnc(CC)cn1)=O)=O 47732,C(=O)(C(O)C(F)(F)F)N1C(C(N2CCC(C(C)C)C2)=O)C(C)C1 47733,CC(C)CC(C(N)=O)NC(c1n[nH]c2c1CCC2)=O 47734,CC1CN2CCN1C(C(=O)NC(C)(C)CNC(=O)CCCN1CCCC1)C2 47735,c1(OC(C)C)ccc2c(c1)CCN(C(=O)C(=O)NCC1CC(O)C1(C)C)C2 47736,CCC(C)(O)C(=O)N1CCN(C2CCCC2NC(=O)C=CC2CCCCC2)CC1 47737,CC1(C)CC(C(=O)NC2CCC2NC(c2cc3cccn3cn2)=O)CC1(C)C 47738,C(=O)(C#CC1CC1)NC1CCN(C(CCN(C)CCO)=O)C1 47739,N1(C(C2N(C)CCCC2)=O)CCN(C(=O)CSc2ccncc2)C(CF)C1 47740,C(CN=c1[nH]c(=NCc2csc(C)c2)[nH]c2c(F)cccc12)(c1ccsc1)OC 47741,c1(C(N2CC(C)C(CNC(C3CC34CCCC4)=O)C2)=O)ccc(F)c2c1OCC2 47742,CC1(C(=O)NCC(C2CCCC2)NC(c2cc(Br)no2)=O)CC(F)C1 47743,N1(C(C(COC)C)=O)CCC2(CCCN2C(c2cncc(OC(F)F)c2)=O)CC1 47744,C1(NC(c2cnc(CC)s2)=O)CC(CNC(c2cn(C)nc2C2CC2)=O)C1(C)C 47745,C1(C(N(C(CNC(c2cc(C)nc(C(F)F)n2)=O)C)C)=O)CCn2nccc2C1 47746,Cn1ccc2cc(C(N3CCC(NC(c4ccc(F)o4)=O)C34CC4)=O)ccc12 47747,C1(NC(c2nc(CC)sc2)=O)CN(C(=O)Cc2cc[nH]c(=N)c2)CC2(CC2)C1 47748,N1(C(C(CCOC)(C)C)=O)CC2(CC(NC(=O)CCCc3cnccn3)CO2)C1 47749,c1(C(=O)NC(C)(C)CNC(C23CCCN2CCC3)=O)ccc2c(c1)NC(=O)CC2 47750,c1(OC)ccc(C(N2CCCC2CN(C(=O)CC2CCCC2C)C)=O)cc1 47751,C1(NC(C(CCC)CNC(=O)CN(C)C)=O)CC(C2CCCC2)C1 47752,C1(C)(C(N2CC(C(C)(C)O)(CNC(CCSCC)=O)C2)=O)CC2CC2C1 47753,C12(C(=O)NC3CC(CC(=O)NCC4CCCCC4O)C3)CCCC1C2(F)F 47754,CC1(C(=O)NC2C=CC(CC(=O)NCCn3cncn3)C2)CCCOC1 47755,c1(OC)cc(C(=O)NCC(C)NC(c2cc(SC)oc2C)=O)c2ccccc2n1 47756,C1(CNC(c2nc(-c3ccco3)n[nH]2)=O)CCN(c2ccccc2)S1(=O)=O 47757,C1(c2n(CCC)nnn2)(NC(c2cccc(Br)c2)C)CNC(=O)C(C)(C)C1 47758,c1(C(N2C(C)CC(NC(c3nn[nH]c3Cl)=O)C2)=O)nccc2ncccc12 47759,c1(C(N2CC(C(C(=O)NCCN3CCC4CC34)OC)C2)=O)c[nH]c2cccnc12 47760,c1(-c2c(NCC)cccc2)cnc(C(=O)OCC)cc1Oc1ccc(Br)cn1 47761,C1(CNC(C2CCC(CC)O2)=O)CCCN(C(=O)Cc2cncnc2O)CC1 47762,c1(C(=O)NC(CC)CNC(=O)CC2CCCOC2)cccc(N)c1C 47763,C1(F)(CNC(C2(C(C)(C)C)CCC2)=O)CCN(C(C2CC(F)(CO)C2)=O)C1 47764,N1(CCC(CC(=O)OCC)(C)C)CC23CCCC2(C1)CN(C)C3 47765,C1(C#N)(C(N2CCC(NC(C(C)n3cncn3)=O)(CF)C2)=O)CC2CCC1CC2 47766,C12(C(N3CC(Cn4cc(C(CCC)=O)nn4)C3)=O)CC3CC(C1)CC(Br)(C3)C2 47767,C(=O)(C(C#N)C(C)C)N1CCC(C(=O)NCc2c(C)scn2)C1 47768,C1(C#N)(C(=O)NC2CC(CNC(C(C)C(F)F)=O)C2)CC2CC2C1 47769,N1(C(C2(CSC)CC2)=O)CCC(CN(C)C(c2cc(C(C)=O)[nH]n2)=O)CC1 47770,CC1CC(C)C(C(=O)NC2CCN(c3nccc(-c4ccccc4F)n3)CC2)O1 47771,N1(C(c2c(C#C)c[nH]n2)=O)CC(=O)NCC1C(=O)NC1CC(c2ncc[nH]2)C1 47772,S(=O)(=O)(c1c[nH]c(C(N2C3CCC2CN(C(c2ccon2)=O)C3)=O)c1)N(C)C 47773,N1(C(C2CCC(CNC(C3C(C)CCCC3)=O)CC2)=O)CC2(CCN(C)CC2)C1 47774,CN1CCC2CCC(C1)N2C(=O)Nc1cccc(Oc2ccccc2)c1 47775,C(c1cc2ccccc2n1OC)=CC(=O)NCC(c1ccc(Cl)cc1)CC 47776,C(=O)(C(C)(C)S(C)(=O)=O)N(C1CCCN(C(=O)C(C)(C)COC)C1)CC 47777,C1(CC)(NC(c2n[nH]cc2C)=O)CN(C(=O)Cn2ccc(C(=O)OC)n2)C1 47778,Cn1ccc2cccc(C(=O)NCC(O)CCNC(C3(C)CC3(F)F)=O)c12 47779,CCC(CC(=O)N1CC(F)CC1CO)NC(=O)C=Cc1cn(C)cn1 47780,CC1CCCN(C(c2csc(CO)n2)=O)C1CNC(C1(C)CC=CC1)=O 47781,c1(OC)ccc(-c2onc(C(=O)NC3CC(CNC(=O)CSC)C3)c2C)cc1 47782,c1(CSC(C(=O)N(CC(CC)NC(=O)C(F)=C(C)C)C)C)ccc(F)cc1 47783,C(CC(C)CN=C(NCC1CC1)N1CCC(NCC(F)(F)F)C1)OC 47784,Nc1cnc(C(=O)NCC2(NC(c3ccc(C4CC4)s3)=O)CCCCC2)cn1 47785,C(=O)(CC(C(F)(F)F)NC(c1sccc1F)=O)NCC1C(C(C)C)C1 47786,c1(C(C)C)oncc1C(=O)NCC1CCN(c2ccccc2)C1 47787,c1(C(=O)NC2(C(=O)NC(C=C)C3CC3)CC2C)cc(CO)[nH]n1 47788,CN1C(=O)OCC1C(=O)NC1CCCCC1NC(C1(Cc2cccnc2)CC1)=O 47789,N1(C(CCCCCC)=O)CC2CCC1C(NC(=O)C(C(=O)OCC)OC)C2 47790,C1(NC(c2cc(C3CC3)nc(Cl)c2)=O)CC1C1CCCN(C(C23CC2C3)=O)C1 47791,C1(C(N2CCC(CC(=O)N(CC(C)C)C(C)C)C2)=O)CC(=O)NC1=O 47792,C(=O)(CC(C)Cc1ccccc1)N(CCNC(c1c(COC)cc[nH]1)=O)C1CC1 47793,c1(OC)ccc(CCNC(=O)C(=O)N(CCO)CC2(C)CCCC2)cc1C 47794,c1(CNC(c2cc(Cl)nc(Cl)c2F)c2n(C)nnn2)cnc2ccnn2c1 47795,C12CC(CO1)C(=O)N2.C(=O)(C(=O)N(CCCOCC)C)NC(CNCCSC)C 47796,N1(C(C(C(C)C)c2ccc(OC)cc2)=O)CCCc2cc(OC)ccc21 47797,N1(C(c2c(C)n(C3CC3)cc2)=O)CC(NC(=O)CCc2ccccn2)C(C)(C)C1 47798,C(=O)(CCCCCF)N(C(C)C(=O)NC(C)(C)CCCO)CC 47799,C12(C(N3CCCC(NC(C(c4cccc(OC)c4)O)=O)C3)=O)CC(N=[N+]=[N-])C1C2 47800,C=CC(CC)CC(=O)NCC1CCC(NC(c2cnn(CC(F)(F)F)c2)=O)CC1 47801,C(=O)(CS(=O)(=O)C1CC1)NCC1C(NC(C(C)Cc2ccncc2)=O)C1 47802,C(CN=c1nc2cccc(Br)c2c[nH]1)C1CCN(C(c2c(C)noc2)=O)C1 47803,N1(C(C2C(C=C)CC2)=O)CC(CO)C2(C1)CN(C(c1cnc(O)c(F)c1)=O)C2 47804,C1(NC(=O)CCc2csnn2)CCCCCC1NC(C1CC2CCC(C1)C2)=O 47805,CCCCCC(=O)NCCCC(C)NC(c1ccnc(N2CCCCC2)n1)=O 47806,c1(NC(C2N(C(C(C)O)=O)CC2)=O)nc(Cl)ccc1F 47807,CC(C)C(CCN(C)C(c1csc(CO)n1)=O)NC(C1(O)CC1(C)C)=O 47808,CC(C)(C)CC(O)CC(=O)NC(CCF)C(=O)NCc1ccc(C(N)=O)o1 47809,C1(C(NNC(C=Cc2c(C)cccc2)=O)=O)C2CCCCCCC12 47810,C(=O)(C(CNC(=O)CC(C)C(F)F)(CC)CC)NCC(CCC)OCC 47811,C1(c2n(CC=C)nnn2)(NCC23CCCC2CCO3)CCC2(CCO2)CC1 47812,N1(C(CC2CC(CC)C2)=O)CCOC2CN(C(=O)COC(C)=O)CC12 47813,CC1COCC(CCNC(NOCCNC(=O)OC(C)(C)C)=O)O1 47814,C(=O)(C1=CC2(CCOC2)C1)N1C(C(=O)NCc2ccc(O)c(F)c2)CC2CC21 47815,c1(C(=O)NCC(CC=C)NC(=O)Cc2ccc(F)c(F)c2)onc2c1CCCC2 47816,CCC(C)CC(C)C(=O)NC1(CNC(=O)C(C)(C)Oc2cccc(Cl)c2)CC1 47817,C(CC(=O)NCC1=CCN(C(c2sc(C#N)cc2Cl)=O)CC1)(C(N)=O)NC(C)=O 47818,c1(C(=O)NCC2N(C(C=C(CC)C)=O)CCOC2)cc2c(C)ccc(C)c2[nH]1 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47889,CN(S(N)(=O)=O)C.c1(C(=O)NCCc2cncnc2)cn(C2CC(C(=O)O)C2)nn1 47890,CCCCCCC(C(=O)NC1(C)CCN(C(=O)C(C)(C)C2CC2)C1)NC(C)=O 47891,c1(C(N2CC3C(CNC(C=C(C)C(=O)O)=O)(C3)C2)=O)ccnc(Cl)c1C 47892,Cc1nc(F)ccc1NC1(c2nnnn2C2CCOCC2)CCN(C2CC2)C1 47893,C1(CNC(C2(OCC)CCCC2)=O)CCCC(NC(=O)COCC(C)C)C1 47894,N1(C(C(C)(C)C2CCOCC2)=O)CC2CCCC(NC(c3cnsc3)=O)C2C1 47895,c1(C(=O)NCC23C(CN(C(c4cn(CC=C)nn4)=O)C2)C3)cccn2cnnc12 47896,CCC(C)C(C)C(=O)N1CC(O)(CNC(c2csc3nnsc23)=O)C1 47897,C(CC(C(=O)NOC(CO)C(C)C)NC(C1CC(C(C)C)C1)=O)=CC 47898,CCC(C(=O)NCC(CNC(=O)C=CCO)OC)Sc1nc(=N)[nH][nH]1 47899,N1(CC(C2CCCCC2)C)CC(=O)N(Cc2ccc(SC(C)(C)C)o2)C1=O 47900,c1(CC)cc(N2CC(C3(C)CC3)C2)n2ncc(Br)c2n1 47901,C1(NC(c2nc(OC)c(F)cn2)=O)CCN(C(=O)CC(=O)NC2CC2)CC1C 47902,C1(C(=O)NCc2c(C)noc2)C2CCN(C(=O)CCC(C)CN(C)C)CC12 47903,C1(NC(C(CC)NC(N)=O)=O)CC2CCC1C(NC(C1CC(CN(C)C)C1)=O)C2 47904,C(C)(C(C)(C)NC(=O)Cc1ccn(C2CCCC2)n1)NC(CSC)=O 47905,CC1CCN(CCC(=O)NCC2C(C)CCN2C(c2cc(C#N)on2)=O)CC1 47906,c1(OC)cc(N(C)C)ccc1C(=O)NCCCCC1CN(C(=O)COC2CC2)C1 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47943,c1(CCC(=O)NCC(C)N(C(c2nc(OCC)oc2)=O)C)c(C)noc1Cl 47944,c1(C(=O)NC(CCCNC(Cc2c(C)cccc2Cl)=O)C)cnc2c(c1)CCC2 47945,N1(C(CSc2ccc(OC)cc2)=O)CCCC(C)C1CNC(c1ccncc1)=O 47946,CN1CCN(C(c2ncncc2F)=O)C(CNC(C2(F)CCOCC2)=O)C1 47947,Cc1nccn1CCCC(=O)NCC1CCN1C(=O)C(F)CC1CCCC1 47948,c1(C(=O)OC)cnc(SC)nc1N1CC2CC1CN2CC.c12ccc(o1)[nH]c2=O 47949,Cc1ncc(NC(=O)C(C)(C)C2CCN(C(=O)C=CC3CCOC3)C2)c(C)c1C 47950,Cc1nc(N(Cc2c[nH]c3c(Cl)cccc23)CC2CNCCO2)c2sccc2n1 47951,c1(CC)cnc(C)c(NC(=O)COC2CCN(C(=O)C=CCOC)C2)c1 47952,C1(CC(C)(C)C)CCN(C(=O)C(C)(C)C2CCN(C(c3cnccn3)=O)C2)C1 47953,N1(C(CCCC)=O)CC(NC(C2(F)CC2C)=O)CC2(CC2)C1 47954,N1(C(C(F)OC)=O)CC(NC(=O)CSc2cc(C)ccc2C)CC(F)C1 47955,c1(CCC(N2C(C(C)NC(C(C)=C3CCCC3)=O)CCC2)=O)ccc(N)c(F)c1 47956,CC(C)CC(CNC(C1CC1C1CCCC1)=O)C(=O)Nc1cc(O)cc(F)c1 47957,c1(OC)ccc(S(=O)(=O)N(c2cc(C3CC3)nn2C)C2CC3CCC2C3)cc1Cl 47958,c1(C(=O)NC2C(NC(=O)CSc3nc[nH]n3)C2)cc(F)cc(F)c1 47959,c1(NCCC(=O)N(CC(C)Cn2cccn2)C2CC2)cnc(C#N)cn1 47960,N1(c2nnc(CC(C)C)s2)CCCC(NC(=O)CNC(C2CC23CC(O)C3)=O)C1 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47978,N1(C(CCc2ccc(C)nc2)=O)CCN(C(=O)CC2CCCC2)C2CC12 47979,c1(C(=O)NC2C(CNC(c3n[nH]c(CC)c3Br)=O)C2)cc(F)cc(Cl)c1O 47980,CON(C)C(=O)CN=c1[nH]c(=NCC2(c3ccsc3)CC2)c2ccc(C)cc2[nH]1 47981,C1(CC(=O)NCC2N(C(C(C)CC3CCCC3)=O)CCC2)COCCOC1 47982,c1(CC)c(C(=O)NCC(C(C)C)NC(=O)CCC(C)(C)C#N)cnc2ncnn12 47983,c1(C(=O)NC2CCC(C)(CNC(C3(CCOC)CC3)=O)C2)nn(C)c(C)c1Cl 47984,C1(CNC(c2noc(CC)c2C)=O)C(C2CC2)CCN1C(c1ccncc1F)=O 47985,C=CCCC(F)(F)C(=O)N1CC(NC(=O)CC(C)(C)C(F)F)C(CC2CC2)C1 47986,N1(C(C(CC)n2cccn2)=O)CCC(C(F)CNC(=O)C(C)(C)F)CC1 47987,C1(SC)CN(C(=O)Cc2occc2C)CC1NC(=O)C(C)CNC(C)=O 47988,C(C(=O)NC1CC(F)(F)C1)(C1=NOC2CC12)N1C(CC#N)CC(F)(F)C1 47989,N1(C(C2CC(SC)C2)=O)CCC(C(C)(C)NC(C2CC(C)C2)=O)C1 47990,c1(NC(C2OCCN(C(C(C=C)O)=O)C2)C)ncc(C)c(C)n1 47991,C1(CNC(CCCCC)=O)CCC(C)CN1C(c1ccc(Cn2cccn2)o1)=O 47992,C1(NC(CCC#CC)=O)CCCCN(C(=O)CCCNC(C)=O)C1 47993,C1(CNC(c2conc2C(F)F)=O)CN(C(c2n[nH]cc2Cl)=O)CC1O 47994,C(=O)(CC(C)(C)SC)NCC(CC=C)NC(=O)CCn1cc(Br)c(C)n1 47995,Cc1cc(C(C)C)ccc1C(=O)NC(C1CCN(C(=O)CC2CCOC2)CC1)C 47996,C1(CC)C(NC(C2CC2CF)=O)CCCN1C(c1ccc(CN(C)C)o1)=O 47997,c1(C(=O)NC(CN(C(c2cc3cccnc3[nH]2)=O)CC)C)cnn2cccnc12 47998,N1(CC)CCOC(C(N2CCCC(CNC(c3ncoc3C(C)(C)C)=O)C2)=O)C1 47999,Cc1cc2ncc(C(=O)NCCC3CC(NC(C4(C)CC4(Cl)Cl)=O)C3)c(C)n2n1 48000,CC1(CNc2nccnc2F)CCN(C(=O)C(c2cccc(F)c2)O)CC1 48001,C(=O)(C1=CCC(C)(C)CC1)NC(CCC)C(=O)Nc1ccsc1C 48002,C=C(Cl)CC(C(=O)NC1CC(C)(O)C1)NC(c1cc(Cl)cn1C)=O 48003,N1(C(c2ncn(C)n2)=O)CC2CCCC(C1)N2C(=O)CC=C(Cl)Cl 48004,CCC(C)C(C(=O)NCc1cnn(C)c1O)N(C(=O)C#CC(C)(C)C)C 48005,Cc1ccc2c(CN3CC4(CC4C(=O)Nc4c(C)cccc4Br)C3)c[nH]c2c1 48006,C1(NC(C2N(CC)C(=O)CC2)=O)CCC12CN(C(c1cnc(S)[nH]1)=O)C2 48007,N1(c2sc(C#N)c(Cl)n2)CCc2sc(NC(=O)C3=CCSC3)cc2C1 48008,CCCCC(CCC)NC(C1(N(C)C(C2CCOCC2)=O)CC1)=O 48009,N1(C(c2c(C)cccc2F)=O)CC(NC(=O)C=CC2CCCO2)CC2(CCC2)C1 48010,c1(C(=O)NC2C(C(=O)NCCCN3CCOCC3)COCC2)cc2occc2[nH]1 48011,N1(C(C2CC(C)(O)C2)=O)CCCCC(C(=O)NC2(C)CC=CCC2)C1 48012,CCC(C(=O)N1CC(C(O)C(=O)CC(=O)NC2CCCC2O)C1)n1cncn1 48013,N1(C(=O)Nc2cccc(Cl)c2)CCC2(CNC(=O)CSc3cccs3)CC2C1 48014,c1(C(c2nnnn2CCCC)NC(C=C)C)nnc(CC)s1 48015,C=C1CCN(C(=O)C(C)CN(C)C(C2(C)CC=CCC2)=O)CC1 48016,c1(C(C)O)ccc(C(=O)NC(C2CN(C(=O)COCP(C)(C)=O)CCO2)C)cc1 48017,N1(C(c2ccc(C)cn2)=O)CC(C)CCC1CNC(=O)C(C1CCC1)C1CCC1 48018,C1(C(N2CC(C(C)NC(C3C(C(=O)OC)C3)=O)C2)=O)CCc2ccnn2C1 48019,C(C(N=c1ccnc(NCCCn2cccn2)[nH]1)C1CCCO1)SC 48020,C1(C(=O)NC2C(C)C2)CC(C)(NC(=O)CC=CC(C)(C)C)C1 48021,CCC(CN=C(NCc1cc2ccccc2o1)N(C)CC1CC1)OC 48022,C(=O)(C(O)C1=CCCCC1)NC1N(C(c2c(C)nc(COCC)s2)=O)CCCC1 48023,c1(C(C)(C)C)ncc(NC(C2CCN2Cc2ccc(Br)o2)=O)cn1 48024,CCCC(CCCNC(=O)COc1ccsc1)NC(=O)C=Cc1c(C)coc1C 48025,N1(C(C2C=C(C)CS2)=O)CCC(NC(C2CCS2(=O)=O)=O)C1C1CC1 48026,CC(C)CC(O)CC(=O)NCc1nocc1C(=O)NCC1(n2ccnn2)CC1 48027,CC1CCC(c2nnnn2C2CCC2)(NCc2cscn2)C1 48028,c1(C(=O)NC2CCN(C(C=C(C)C(C)C)=O)C2C)cc2cccc(C)n2n1 48029,c1(CC(N2C3(CNC(=O)CCC4CCC4)CCC3CC2)=O)cc(F)c(F)cc1F 48030,n1(CC(=O)NCC2C(NC(c3c(C)nc[nH]3)=O)C2)sc2ccccc2c1=O 48031,c1(C(=O)NCC2CN(C(c3ccc(SC)o3)=O)CC2C)cc(N(C)C)ccc1Cl 48032,N1(C(C2CC(C#N)(OC)C2)=O)CC(C(=O)N(CCC(F)(F)F)C)OC(C)C1 48033,C1(CC(C)C)CCN(C(C2CCN(C(=O)CCc3cn(C)cn3)C2)=O)C1 48034,C1(NC(C2(CCC=C)CN(C(c3cc[nH]c3)=O)C2)=O)CCn2cncc2C1 48035,c1(CC(=O)NC(C(=O)N(CC)Cc2ccncc2)C2CCOC2)cncnc1O 48036,C1(C(=O)NCCC(=O)NCC#C)COC2(C1)CN(C(c1cnc(OC)nc1)=O)C2 48037,c1(C(=O)NC2CC3CN(C(C(COC)(C)C)=O)C2C3)c(C)nc2sc(C)nn12 48038,N1(C(CC2N(C(C3=CCCCC3C)=O)CC(C)(C)C2)=O)CCCC2C(=O)NCC12 48039,c1(C(N2C(CC)C(O)CC2)C(=O)NCCC2(C)CC2)cc2c(s1)CCOC2 48040,C1(CCC(=O)OC)(OC)CCNCC1.N1(C)CCC1(C)C1CCCCC1 48041,C(=O)(C(F)C(C)CNC(c1ccc(O)cc1)=O)NCCCCOC 48042,C12(CNC(CCOC)=O)CCC1CCN2C(=O)C(=Cc1ccco1)C 48043,C(=O)(CC(O)C(C)(C)C)N1CCC(NC(Cn2c(C)ccn2)=O)C1C 48044,N1(C(C2N(CC)CCC2)=O)CCC(C)(CNC(c2sncc2C)=O)C1 48045,C1(CCOC)(NC(=O)CCC2CC2)CCN(CC=C(Cl)Cl)CC1 48046,c1(OCC)c(OC)cc(CNCCCc2ccc(OC)cc2C)cc1Br 48047,c1(C(N2C(CN(C(CC(C)C3CC3)=O)C3CC3)CCC2)=O)c(C2CC2)cnn1C 48048,C1(C(=O)NCCN(C(=O)COc2cccc(Cl)n2)C)CCN(CCO)C(=O)C1 48049,C(CC(O)CC(=O)N(C)CCN(C(=O)C(C)(F)CC)C)SC 48050,[N-]=[N+]=Nc1ccnc(CNC(=O)CC2CC(O)CN2C(=O)OC(C)(C)C)c1 48051,c1(C(=O)NCCCC(CCC)NC(c2nc(Cl)oc2C)=O)cnc2ncccn12 48052,Cc1nc2ccc(C(=O)NC3CC(CNC(=O)CC4CCCC4)C3)cn2n1 48053,C(C)(CNC(c1ccn(C)c1)=O)(CC(C)C)NC(Cc1nc(C(C)OC)sc1)=O 48054,N1(C(C2CC(=C)CN2C(=O)Cc2cc(Br)ccc2Br)=O)CCC(O)C(C)(CO)C1 48055,c1(CC)nc(C)oc1C(N1CC2C(N(C(=O)C(CC)SC)C)C2C1)=O 48056,Cc1cc2c(C(N3CCC(CNC(=O)CSC(F)F)CC3)=O)cccc2[nH]1 48057,C1(C)(C(=O)NC2CCN(CCC)C2)CCCN(c2cc[nH]c(=N)n2)C1 48058,c1(N2CC(CNC(C(CC)SC)=O)OCC2)cc(C)c([N+](=O)[O-])cn1 48059,n1(CC)c(N2CCOC(C)C2)nnc1C1(NC(C)(C)C)CC1 48060,Cc1nc(C(=O)NCC(C)(C)CN(C)C(C2CCSC(C)C2)=O)cn1C 48061,CC1(F)CN(C(c2cccc([N+](=O)[O-])c2)=O)CCN(C(c2cccc(=O)o2)=O)C1 48062,C1(CC=O)C(=O)N(C)C(C)(C(=O)NCCOC(F)F)C1CC 48063,Cc1ncc(N)cc1C(=O)NC1COCC1NC(=O)Cc1cc(C2CC2)nn1C 48064,Cc1cccc(Br)c1S(=O)(=O)NCCCc1ccc([N+](=O)[O-])cc1 48065,CN1C(C(=O)NC2CC(C)(NC(=O)CC(C)(C)C#N)C2)CCS1(=O)=O 48066,c1(NC(c2n(CCC)ncc2)=O)ccc(NC(=O)C(C2(O)CCCC2)F)cc1C 48067,Cc1nsc(C)c1C(=O)NCC1CCCCC1NC(C1(C2CC2)CCC1)=O 48068,C(CC(=O)N(C(CO)CO)C)(C(F)F)NC(c1cc(C)n(C)n1)=O 48069,C1(O)(CCNC(C2(CCC)CCC2)=O)CCN(C(=O)Cn2ncc(Cl)c2C)C1 48070,c1(C(C2CCCC2)OC)nc(-c2cccs2)nn1-c1ccnc(F)c1 48071,C(=O)(C(F)(F)CC(C)C)NC1(COC)CCN(C(=O)Cn2cc(Cl)cn2)C1 48072,C1(NC(N(C2CCN(c3ncccn3)C2)C)=O)CCCOC1 48073,C(CS(=O)(=O)CC(=O)N(C)CC1CCCCN1C(c1coc(C(F)F)n1)=O)OC 48074,N1(C(C2C(CC)C2)=O)CC(CNC(c2cccc(SC)c2N)=O)CC12CCC2 48075,c1(CN(C)C)cnc(O)cc1C(F)(F)F.C12CC(C1)NC2=O 48076,C(C(C)(C(=O)NCC1(O)CN(C(=O)C=Cc2ccncn2)C1)OC)OC 48077,N1(C(C2(C)C(C)OCC2)=O)CC(C2(NC(c3cnnn3C)=O)CC2)C1 48078,C1(C(N(CCC(=O)NC2CC2CSC)CC)=O)CC=CCC1 48079,CCC1=NOC(C(=O)N(CC(C)NC(c2cccc(C(C)(F)F)n2)=O)CC)C1 48080,N1(C(C(C2CCOCC2)C)=O)CCC(C)(C(=O)Nc2cccc(C(F)F)c2)C1 48081,Cc1nc(CC(N2CCC(CO)(NC(C3CCC(=O)O3)=O)C2)=O)c(C)s1 48082,C1(CC)CN(C(c2c(C)cnn2C)=O)CCN1C(c1ccc(SC)s1)=O 48083,c1(CC(C)C)c[nH]c(C(=O)N(C)CCNC(=O)CC2C=CCC2)c1 48084,c1(C(N2CCC(N(CCC)C(C3CC=CC3)=O)C2)=O)cc(CC)nc(O)c1 48085,O=C(C(O)C1=CCCCC1)NCC1CCN1C(=O)Cc1ccc(C(F)F)cc1 48086,CCCC(O)CC(=O)NCC(C1CCCC1)NC(=O)C(c1cccc(F)c1)C 48087,Cc1ncncc1C(N1CC(NC(C2OCCC2C)=O)C(C)C1)=O 48088,C(N=c1[nH]c(N2CC(C(F)F)C3(CCC3)C2)nc2c1COC2)c1c(C)cncc1 48089,c1(C(=O)NCC(=C)CCNC(=O)CCC=CBr)c(C)[nH]c2ccc(OC)cc12 48090,c1(CC)c(C(N2CCC(C3CCCN3C(c3[nH]ncc3C#N)=O)C2)=O)cnn1C 48091,c1(C2(NC(C(C)c3ccco3)=O)CC2)ccc(C(=O)O)cc1 48092,CC1CCCN(C(=O)C=CC(C)(C)NC(C23CC2CNC3=O)=O)C1CO 48093,N1(C(C)C)C(=O)COCC1C(N1CCC(CNC(=O)C2=CCOCC2)C(C)C1)=O 48094,C(CCCCC(=O)NC(c1cnn[nH]1)C)N(C(c1cccc(C)c1)=O)C 48095,N1(C(c2cnc(SC)s2)=O)CC(C)C(NC(=O)COc2cccnc2Cl)C(C)C1 48096,N1(C(C(CC)C2CCOCC2)=O)CCN(C(=O)CCCCCSC)CC2(CC2)C1 48097,N1(C(C#C)=O)CCc2c(C(=O)Nc3ccc4nc(Cl)sc4c3)n[nH]c2C1 48098,Cc1cc(F)sc1C(=O)NCC(C)NC(=O)Cc1cccc(OCC(F)(F)F)c1 48099,C1(CC(N2CC(CCNC(=O)CCn3cccc3)OCC2)=O)CCCCCCC1 48100,N#Cc1cn(CC(=O)NC2CN(C(C3NC(=O)C4CC34)=O)C2)c(=O)nc1O 48101,c1(C(=O)NC(CN(C(C)C)C)C)ccccc1NC(=O)C(C)NC(N)=O 48102,C1(c2n(CCC)nnn2)(Nc2nn(C)c(C)c2Cl)CCN(C(=O)C(F)(F)F)CC1 48103,C1(NC(CC(c2ccc(F)cc2)C)=O)CCCN(C(C2COC2)=O)CC1 48104,c1(C(N2C(C(C)NC(c3c(C)ncnc3)=O)CCCC2)=O)cccn2cncc12 48105,C(=O)(CCCCCN(C)C)NC1CC(F)(CNC(c2ccnc(CC(C)C)n2)=O)C1 48106,Fc1cccc2nc(N3CCC4CC4C3)[nH]c(=NCC3(CCO)CCC3)c12 48107,c1(C(N(CCC(C)NC(C(C(C)C)O)=O)C)=O)ccc(F)c(C#N)c1 48108,c1(C(=O)NCC2CCCN(C(C3COCCO3)=O)C2)ncc(C2CC2)cc1F 48109,Cc1ccc(C(=O)NC2CC(NC(C3(c4ncco4)CC3)=O)C23CCC3)nc1O 48110,c1(C(=O)NCC(N(C(CC=C=C)=O)C)C2CC2)cccc2c1OCCN2 48111,C1(CNC(C2CC(CC)OCC2)=O)CC2CCC1N2C(C1CNC(=O)N1)=O 48112,Cn1cnc2sc(C(=O)NC3CCCC(NC(=O)Cc4cc[nH]n4)CC3)cc12 48113,c1(COC)c(C(=O)NC2(C)CC(NC(c3ccnn3C)=O)C2)sc2ccccc12 48114,C1(OC)CCN(C(c2c(C(=O)OCC)[nH]cc2C)=O)C(c2ccccc2)C1 48115,CC1CC(C(=O)NC2CCCCC2NC(c2cn(C3CCOC3)nn2)=O)CN1C 48116,C(=O)(C(O)C(F)(F)F)NCCC(CNC(c1n(CC)ncc1)=O)O 48117,N1(C(CC2C(NC(C(C(C)(F)F)F)=O)CCCC2)=O)CCCC12CCOCC2 48118,c1(CCC(=O)NC(CN(CC)CC)C)ccc(CO)cc1.C1(C)(C=O)CC1(F)F 48119,c1(CCC)ccc(C(c2nnnn2C2CC2)NCC2CCCOCC2)cc1 48120,C1(C(=O)NCCCC(C)NC(C(C2CCCCC2)OC)=O)CN2CCCN1CC2 48121,C12(N(c3ccccc3)C(=O)CCOC(C)(C)C)C(CC1SC)OC2=O.CO 48122,c1(C(=O)NC(C(CO)NC(C(CSC)C)=O)C)ccc(Br)c(SC)c1 48123,C1(C(N(CCCCN(C(C(C)C#N)=O)C)C)=O)CCn2cncc2C1 48124,N#Cc1ccnc(C(=O)NC2CCN(C(C3CCCN3CC(F)(F)F)=O)C2)c1F 48125,c1(C(C)N(C)C(C2(C(C)(C)C)CCNC2)=O)ccc(F)cc1 48126,Cc1ncc2cc(C(N3CC4CC(NC(=O)CCc5csnn5)C3C4)=O)ccn12 48127,C1(C2CC2)(CNC(C(N2CCC(C)CC2)=O)=O)CCN(C(C2(C)COC2)=O)C1 48128,C1(CNC(C2C(CCC)CCC2)=O)CN(C(=O)C=Cc2cnc(C)s2)CCCO1 48129,c1(C(C(=O)NCC(CC)(C)NC(=O)CCC=CC(C)C)C)ccc(OC)cc1C 48130,N1(C(C2CCC(=O)NC2)=O)CCOC2CN(C(c3cnc4ccccn34)=O)CC12 48131,c1(C(=O)NCC2OCC(CNC(CCC)=O)C2)cc2cccc(Br)c2cn1 48132,N1(CCC)CC2C3CCC(C2C1)N(c1nc(Cl)nc2[nH]ccc12)C3 48133,N1(C(CC(C)C)=O)CC(C(N2CCCCC2C2(O)CC2)=O)C(C(C)C)C1 48134,C1(C)(C(=O)NC2CC(CCNC(C3(OC)CCC(C)C3)=O)C2)C(C)(C)C1(C)C 48135,Cc1cccc(CC(=O)N(C2CCC(NC(=O)Cc3nccn3C)C2)C)c1 48136,C(=O)(C(F)CC(C)(C)NC(c1cc(C)n(C)c1C)=O)N(CC(=O)OCC)C 48137,C(=O)(C(CC(C)C)C(C)C)NC1CC2(C(C(N(CCOCC)C)=O)C2)C1 48138,C1(CC(=O)NC(CNC(C(c2cnn(C)c2)C)=O)(C)C2CC2)CNC(=O)C1 48139,c1(C(N2CC(C(=O)OC3CCC(CCCC)CC3)C2)=O)c(F)ccc(CC)c1F 48140,N1(C(CCC(=C)C)=O)CCC(NC(=O)CN2CCC(C(N)=O)CC2)CC1C1CC1 48141,c1(C2CCCN(Cc3ccn(CC)n3)C2)cccc(NC(C2(CSC)CC2)=O)c1 48142,C1(CCC#C)CCCN1C(=O)C(CNC(c1[nH]nnc1C)=O)N(C)C 48143,Cc1nc(S)nc(C)c1CCC(=O)NCC1(NC(C2CCN(C)C2=O)=O)CCC1 48144,C1(C(CC)C)CCN(C(=O)COC2(C)CN(C(=O)C(O)CC)C2)CC1 48145,C(=O)(C(C)C(C)COC)NCCOCCNC(C1(CC)CC(F)(F)C1)=O 48146,N1(C(CNC(CC)=O)=O)CC2CC(NC(c3ccn(C4CCCC4)n3)=O)C(C2)C1 48147,N1(C(C)=O)CS(=O)(=O)CC1C(=O)NCC1CN(C(=O)Cc2cn3ccsc3n2)C1 48148,Cc1ccncc1C(=O)NCC#CC(=O)NCc1ccco1 48149,N1(C(C(F)OC)=O)CCC2CCN(C(C3CN4CCN3CC4)=O)CC12 48150,c1(CC)nn(C)c(C(=O)NCC2CN(C(c3ccc(SC)o3)=O)CCC2C)c1Cl 48151,C1(C(=O)NCCC(=C)CNC(C2CC(F)C2)=O)CC(C2CCOCC2)=NO1 48152,c1(C(=O)OC)cc(=NCC2CCC(NC(c3cc(C(C)(C)C)on3)=O)C2)[nH]cn1 48153,C1(CNC(c2cnnc(O)c2)=O)CC2CCCCC2N1C(c1ncc(F)cn1)=O 48154,c1(C(=O)Oc2c(C(=O)OC)scc2NC(=O)C(=O)NCC)ccc(F)c(OC)c1 48155,C(CCCCCC(=O)Nc1cncc(C#N)c1)NC(C1(OCC)CCOC1)=O 48156,CCC(CC)C(=O)NCC1C(Cn2cc(-c3cnn(CCOC)c3)nn2)C1(F)F 48157,C#CC1(C(N(C)C[Si](C)(C)C)=O)CCN(C(=O)CCC2CCCO2)C1 48158,N1(C(C2(CC#C)CCCCO2)=O)CC(NC(=O)CCCC2CCCC2)CC(F)C1 48159,N1(C(Cc2c(C)con2)=O)CC=C(CC(=O)N2CCC3CC23C)CC1 48160,c1(C(n2nccn2)C)nnc(N2CCN(CC)CC2)n1Cc1ccc(NC)cc1 48161,c1(C(=O)NCC2N(CC(=O)NC(N)=O)CCC2)ccn2ccnc2c1 48162,C1(C(C(=O)N(CCCC)C2CC2)C)CCCN(C(=O)C(OC)OC)C1 48163,c1(OC)ccc2c(=NCc3csc(Br)c3)[nH]c(NC3CCOC(C)C3)nc2c1 48164,c1(C(N2CC(NC(C(C3CCOCC3)OC)=O)C(F)C2)=O)cc(N)ccc1SC 48165,C1(c2nnnn2C)(NCc2n(C)nc(-c3ccccc3)c2)CCC(N(C)C)CC1 48166,c1(C(N2CC(NC(C3C(C)C3C)=O)C3(C2)CC3)=O)cc2cc(F)ccc2[nH]c1=O 48167,c1(C(=O)NC2CN(c3ccnc(C4CCCC4)n3)C2)cc(F)c(OCF)c(F)c1 48168,Cc1ncccc1C(c1nnnn1CC1CC1)NC(c1ccccc1)C(N)=O 48169,Cc1cc(CC(=O)NC(C)C(C)(C)NC(=O)Cc2csc(Cl)c2)n[nH]1 48170,N12CCC3(CC(C3)C(=O)NC(CC=C)CC1=O)C2.c1(C2(CC)CC2)cc[nH]n1 48171,N1(C(c2ccn(CCNC(CCN(CCC)C)=O)c2)=O)CCC12CCC(C)CC2 48172,C1(F)(CNC(c2n(CCC)ncc2)=O)CCN(C(C2CC3CC3CC2C)=O)CC1 48173,c1(C(C)C)nc(=N)[nH]c(=NCCCCNC(=O)CN(C2CCSC2)C)[nH]1 48174,N1(C(C(C)n2ccnn2)=O)CC2(CCC(CNC(=O)CCF)O2)C1 48175,C(=O)(C1CCCc2nnn(C)c21)N(CCCNC(=O)CCCC1CCC1)C(C)C 48176,C1(CNC(c2on(C)c(=O)c2)=O)(CO)CCN(C(=O)Cc2cnns2)CC1 48177,C(=O)(C1=NOC(C)C1C)NC1C(OC)CN(C(=O)CCCC2CCCCC2)C1 48178,c1(C(N2CC(CNC(=O)C=CC3CCCCCC3)C2)=O)ccc2nnn(O)c2c1 48179,C1(C(=O)NCCNC(C2(F)C3CCCC23)=O)CC2(C1)CC21CCC1 48180,CC(CNC(=O)C(CCC1CCC1)NC(=O)COc1ccccc1)C(F)(F)F 48181,C1(C(=O)NC(C)CN(C)C(c2cnncc2O)=O)CN(C)CCN(C)C1 48182,CC1=C(C(=O)NCC2CCC(NC(C3OC(C)CC3C)=O)C2)CCCO1 48183,Cc1nc(Cl)nc(N2CCCC(C(C)NC(=O)C=Cc3ccncc3)C2)c1F 48184,CCS(=O)(=O)CC(=O)N1CCOC(CN(C(=O)CC2(C)CC(F)(F)C2)C)C1 48185,C1(C(=O)NCC2CCN(C(=O)CN3CCCCC3)C2)CCC2(CC1)OCCO2 48186,Cn1cncc1C=CC(=O)NCCN(C(C1CC1c1cccnc1)=O)C1CC1 48187,C(=O)(C1CCS(=O)(=O)c2ccccc21)NCC(CNC(Cc1ccc(C)s1)=O)C 48188,Cc1ncccc1C(=O)NCc1cc(C(N2CCC(C(C)(C)O)CC2)=O)ccn1 48189,N12C(=O)CCC(C1=O)N(C)CCNC(=O)C2=O.N1(CC)CC(C)(SC)C1=O 48190,c1(C(=O)NC2C(NC(C(C)(C)n3ccnn3)=O)C2)cc(F)c(Cl)cc1Cl 48191,N1(C(CC(C)c2cccnc2)=O)CC2CC2(CNC(=O)CN(C)C(N)=O)C1 48192,CCCCC(CC)CC(=O)NCC1CCC2CN(C(C3CSC3)=O)CCC2C1 48193,C1(O)(C(C)NC(=O)COC2CCCC2)CN(C(=O)CCc2nccs2)C1 48194,CC(C)C(O)C(=O)NC(C)CCNC(=O)CCC1CCCC1 48195,C(C)(CCC(=O)N(CCCNC(=O)Cn1nc(C)cc1C)C1CC1)SC 48196,C(C(CC(C)C)C(=O)N1CCN(C(c2cc(CO)c(CO)o2)=O)CC1CO)OCC 48197,C1(O)(CNC(c2nc(CNC(CS(=O)(=O)NC)=O)oc2)=O)CC2CCC1O2 48198,C12(NC(=O)CSCc3cscn3)CCCN(c3ccn4nccc4n3)CC1C2 48199,Cc1cccc(CNC2CCN(C(c3cc(C(=O)O)ccc3F)=O)C2)c1C 48200,n1(CC(=O)NC2C(SC)CN(C(C3(CO)CCCC3)=O)C2)nc(C)c(Cl)c1C 48201,CC1CC(C(N2CCCCC2C2CCOC2)C(=O)NC2CCOCC2)CC(C)C1 48202,Cc1nc(O)sc1C(N1CC(CC(=O)NC(C)Cc2nncn2C)CC1C)=O 48203,N1(C(CNS(NC)(=O)=O)=O)CCCC2CCN(C(c3nocc3Cl)=O)CC12 48204,c1(C(=O)NC2CCN(C(c3cscc3C3CC3)=O)C2)ccc(SC(F)(F)F)nc1 48205,c1(C(=O)Nc2scc(COC)n2)cc(Br)cnc1C(F)(F)F 48206,C1(NC(CC=CC)CO)CCOC2(CCOCC2)C1 48207,N1(C(CCC(=C)C)=O)CC(CNC(=O)CCCC)CC12CCOCC2 48208,Oc1nc2ccccc2cc1NCCN1CCCC1 48209,N1(C(C(N2CC(C)CC(C)C2)=O)=O)CCn2c(cnc2C(N2CCOCC2)=O)C1 48210,N1(CCC)C(=O)CCC1C(=O)NC(CNC(=O)C=C1CCSCC1)C1CCC1 48211,CCC1(C(=O)NCC(CC)NC(c2ccsc2C)=O)CCCc2ccccc21 48212,Cc1nn(CC(=O)NCC2CCC3(CN(C(=O)C(C)CF)C3)O2)c2ncccc12 48213,C1(C(=O)NC2C(CNC(c3cnoc3C3CC3)=O)C2)CC2(C1)CC2(F)F 48214,c1(C(=O)NCC(CNC(C(C(C)(C)C)SC)=O)F)cc(Cl)c2n[nH]cc2c1 48215,Cc1cc(Cl)cc(C(N2CCOC(CN(C)C(c3ccc(F)s3)=O)C2)=O)c1N 48216,CC1CCC1C(=O)NC(C(=O)NCC=CCl)C1CCCC1 48217,c1(C(N(C)CC2CCN(C(C(C)(C)OC(C)=O)=O)C2)=O)ccc(Br)c(C)n1 48218,CCCCCC(C)(C)C(=O)NC1CCOC(CNC(C2CCC2COC)=O)C1 48219,c1(C(=O)NCC2N(C(C(COC)(C)OC)=O)CC2)cc(Br)cc(OC)c1O 48220,c1(OC)ccc(F)cc1CNC(=O)NCC1CC2(CCC2)CN1 48221,Cc1ccc(CCC(=O)NC2CN(C(=O)COC3CCCC3)C(C)(C)C2)cc1Cl 48222,C1(C(=O)OC)CCCC1NC(=O)NCCNC(c1sncc1C)=O 48223,Cc1cccnc1C(=O)N(CC(O)CN(C)C(c1cc(CC(C)C)nn1C)=O)C 48224,CC1(C(=O)Nc2cc(O)ncn2)CCN(C(c2ccccc2C2CC2)=O)CC1 48225,C1(C(N2CCC(CO)CC2)=O)CC2CC2N1Cc1cccc(-c2ccccn2)c1 48226,c1(C(=O)NC(CC)CNC(c2ccncc2N)=O)cc(S(=O)(=O)NC)oc1C 48227,C1(C(=O)NC2(COC)CCC2)CC(F)(CNC(CN(CCC)C)=O)C1 48228,N1(C(C(C)(C)C)=O)CCCC(F)(CNC(c2cccc(C3CC3)c2Cl)=O)C1 48229,c1(CCC(=O)NCCCCNC(C2CCC2C2CC2)=O)c(Cl)cccc1Cl 48230,c1(C(=O)NC2CC(NC(C(C)C3(O)CCC3)=O)C23CCC3)cc2c([nH]1)CCCC2 48231,N1(c2ccc(C#C)cc2)CCC2C(CCN2S(=O)(=O)CCCCCCC)C1 48232,C(=O)(CS(=O)(=O)Cc1cccs1)NCCOC1CCN(C(C(CC=C)C)=O)C1 48233,C1(C=C)(C(N(C(C(=O)NC(CCSC)C)C)C2CC2)=O)CCCCC1 48234,c1(CN(C(C2CC(=O)C2)=O)C2CC2)c(F)cccc1F 48235,N1(C(=O)CN2CC3CC3C2)CC2CCCN(C(C3CCC(F)C3)=O)C2C1 48236,CN1CC(C(=O)NCC2CC2CNC(C2(C(F)F)CC(F)(F)C2)=O)NC1=O 48237,C(C(=O)NNc1ccc(S(=O)(=O)N(C)C)cc1)(C(C)(C)C)n1cc(COCC)nn1 48238,C12(CNCC3CNCC(C(F)(F)F)O3)CCCN(CCC1)C2 48239,N1(C(C2C(C)CCC2)=O)CC2CCC1CC2NC(c1cnn(C)n1)=O 48240,c1(C(=O)NC2CN(C(c3cnsn3)=O)C3(CCC3)C2)cc2ccnc(Cl)c2s1 48241,Cc1nc2cc(C(=O)NCC3(NC(C4CCN(CC(F)(F)F)C4)=O)CC3)[nH]c2s1 48242,c1(C(=O)NCCCCN(C(c2cc(C(C)=O)on2)=O)C)cc(C)c(Cl)cn1 48243,c1(NCCN(C(C2(F)CCS(=O)(=O)C2)=O)CC)ncc(C#N)cc1F 48244,N1(C(CC(C)c2cnn(C)c2)=O)CCCCC1CN(C(=O)C1=CCOC1)C 48245,n12ncc(c1N)C(=O)NC2.c1(NC(C=CC=CC)=O)cnn(CCOC)c1 48246,CCC(CNC1(c2nnnn2C2(C)CC2)CCC(SC)C1)(CC)SC 48247,N1(C(C2N(CC#C)CCC2)=O)CCC(NC(C2C(C)OC(C)C2C)=O)C(F)C1 48248,CP(C)(=O)c1ccc(C(N2CCC(CNC(=O)C3=CCCCC3)C2)=O)cc1 48249,c1(C(=O)NCC2(NC(C3COC3)=O)CC2)cnc(C2CCC2)s1 48250,c1(C(N2CC(C(C)NC(c3c(OC)cnc(Cl)c3)=O)C2)=O)ccc(F)c(C#N)c1 48251,C1(C(N(CCN(C(CCN(CC)CC)=O)CC)CC)=O)CCCCC(F)(F)C1 48252,c1(OCC)ccccc1COCC(O)CN(C)Cc1cccnc1-n1cccn1 48253,N1(C(=O)NCC2(CO)CC2)CCCC2(NC(=O)CCc3cccc(F)c3)CC2C1 48254,c1(C(=O)NC2CN(C(c3coc(Cl)n3)=O)CC23CC3)ccc2cccnn12 48255,c1(C(=O)NC2CCCN(C(CC(CCC)O)=O)C2)cnc2c(C)c(Cl)ccc2c1 48256,CC(CCNC(=O)CNS(N)(=O)=O)CCNC(=O)C(C)(C)C1CCOCC1 48257,C1(C(N(C2CC2C)C)=O)CC12CCN(C(=O)Cc1cccc(Br)c1)CC2 48258,CC(CC(F)(F)F)C(=O)N1CC(CCNC(c2cc(=O)cc(Cl)[nH]2)=O)C1 48259,C1(NC(C(C)OCCC=C)=O)CN(C(C2(C#N)CCCC(=O)C2)=O)CC(C)(C)C1 48260,C1(C(N2CCCCCC2CNC(=O)C(F)(F)c2cncs2)=O)CCCCC1(F)F 48261,c1(C(N(CC(C)O)CCNC(c2c(C)n(C)nc2)=O)=O)cccn2c(C)cnc12 48262,CC1(NC(c2csc(CC(F)F)n2)=O)CN(C(=O)CC2CC3(CC3)C2)C1 48263,N1(C(C2C(CC(C)C)C2)=O)CC2CN(C(=O)Cn3ccccc3=O)CCC12 48264,C1(CNC(C(CC)(CC)CO)=O)CCN(C(C2CC2C(=O)OC)=O)CCC1(F)F 48265,CCCCCCC(C)C(=O)N1CC2CN(C(c3cc(Cl)cc(OC)c3N)=O)C2C1 48266,Cc1nc[nH]c(=NCC(C2CCCCC2)NC(c2c(C)nn(C)c2C)=O)c1C#N 48267,c1(CC(N2CC(NC(CC(C)(C)O)=O)C(C)(C)CC2)=O)ccc2cccnc2c1 48268,C12(CNC(CN(C3CCSC3)C)=O)CCCC1N(C(=O)CC1OCCO1)CCC2 48269,N1(C(C(COC)COC)=O)CCN(C)C(C(=O)NCCCN(C)C(C)=O)C1 48270,CCCC(CC(=O)N(CC(O)C1(Cl)CC1)C)NC(=O)C(C)NC(=O)C1CC1 48271,N1(C(c2c(C)oc(Cl)n2)=O)CC(NC(=O)C=Cc2cncnc2O)C(N=[N+]=[N-])C1 48272,CCCC(C)CCNC(=O)C(C1CCN(C(c2ccccc2O)=O)CC1)C 48273,C1(N(C)C(N)=O)CCCC(N(C(=O)CN2CCC(C)(C)C2)C)C1.C1(=O)CCN1 48274,N1(C(C2N(C)CC(O)C2)=O)CCN(C)C(CNC(=O)COC2CCC2)C1 48275,c1(C(=O)NC2CC(C)N(C(=O)CC3CC=CCC3)C2)cnc2cccnc2c1 48276,Cc1cc(NC(C2CCCCCC2)C)ncc1C(F)(F)F 48277,C(=O)(CC(C1CC1)C1CC1)NCC1CCCCO1.C12CC1C(=O)NC2C 48278,C1(C(=O)NC(C=C)(C)C)CCC(C2CC2)N1C(c1cc(Cl)cs1)=O 48279,N1(C(c2cn(CC)nn2)C(=O)NCC2CCCO2)CC2(CO)CC2(C(F)(F)F)C1 48280,C1(C(=O)NC(C(=O)NC2CCN(CCC)C2)CC)CC12CCCCC2 48281,N1(C(C=C(CCC)C)=O)CCC(C2CC2)C1CNC(=O)Cc1c(C)cccc1C 48282,N1(C(c2c(C)nc(CC)s2)=O)CC(C2CN(C(C34CCC(O)C3CC4)=O)C2)C1 48283,c1(-c2c(C(N3CCOC4CC34)=O)n[nH]c2)cccnc1-c1ccccc1 48284,C(=O)(C(C)CC(C)(C)C)N1CC(F)CC(NC(c2ccc(OC)cc2C)=O)C1 48285,C#CCC(CC(=O)NC(CC)C(C)(C)C)NC(C1CS(=O)C1)=O 48286,c1(CNC(C=C2CCC(C)CC2)=O)nc2c(s1)CCN(C(=O)Cc1cocn1)C2 48287,C(CC1CCC1)(C(=O)NC1CCC1)N(CCCF)C 48288,N1(CC(=O)N=c2cco[nH]2)CC2CCN(C(c3nc[nH]c3C(F)(F)F)=O)CCC2C1 48289,C12(C(=O)NCC(CNC(c3ccn4ncnc4c3)=O)O)CCC(O)(CC1)CC2 48290,C1(CCC(=O)NC(C#C)C2CCC2)CCCN(C(=O)CC(O)c2ccccc2)C1 48291,C1(CNC(C(C2CC2)OC)=O)C(C)CCCN1C(=O)C(=Cc1ccc(C)cc1)C 48292,C1(NC(c2c(C)ccs2)=O)CC2CC(NC(=O)C(O)C(C)C)CC2C1 48293,C1(NC(c2nn(C)c(C(N)=O)c2)=O)CC2CCC(C1)N2C(=O)C(O)C1CCC1 48294,C1(NC(N2CC(CCNC(c3ccccc3)=O)C2)=O)CCC2C(CC1)C2(F)F 48295,N1(C(c2cc(C)ncn2)=O)CCC(C2CCN(C(c3ccccc3C)=O)C2)C1 48296,C(=O)(CC1=CCN(C(=O)CCOCC(C)C)CC1)NC1(C(=O)NC)CCC1 48297,C1(C(=O)N=S(C)(=O)CCOC)N(C(=O)OC(C)(C)C)CC12CCCC2.C(=O)OC 48298,Cc1n[nH]c(C)c1SCC(N1CCCC(CN(C(=O)C(C)CC2CCC2)C)C1)=O 48299,C1(CNC(Cn2nc(C)oc2=O)=O)CC(C(=O)NCC(C)(C)C#N)=NO1 48300,CCC(O)C(C)C(=O)NC12CC(C1)N(C(=O)CCc1cncnc1)C2 48301,c1(CC(=O)NC2CCC(NC(Cc3c(Cl)cn(C)n3)=O)C2)cc(F)ccc1Cl 48302,S(=O)(=O)(c1cc(Br)cc2c1OCC2)NS(CC1(Cc2ccc(C)cc2)CC1)(=O)=O 48303,Cc1c(C(=O)NC(CNC(C2CC3(CCC3)C2)=O)C(C)C(C)C)cc(O)cc1N 48304,CC(C(=O)N1CCCN1C(=O)Oc1ccccc1C(F)(F)F)C1CCCNC1 48305,C(=O)(C1CCCc2c[nH]nc21)N1C(c2nnc(-c3ccc(P(C)(C)=O)o3)o2)CCCC1 48306,C12(CNC(C3C(OC)CCC3)=O)CCC1CN(C(=O)Cc1cccc(F)c1F)C2 48307,c1(N2CCCN(CC=C)CC2)nc(=NC)nc(N2CCn3cncc3C2)[nH]1 48308,C12(C(=O)NCCCOC(=N)O)CC(CN1C(=O)CC1CCOC1)C2 48309,O=C(C#CC1CCOCC1)NCC1CN(C(c2ccc(C(F)F)o2)=O)CC1(F)F 48310,c1(C(=O)NCC(C2CC2)NC(C(C(=O)OCC)OC)=O)cc(S(C)(=O)=O)oc1C 48311,C1(CC)CN(C(=O)Cc2cc(C)n(C)n2)CCC1CNC(=O)C(CC)(CO)OC 48312,c1(NCC2C(c3n(C)ncc3)C2)ccc(S(=O)(=O)N2CCOCC2)c(Br)c1 48313,CCCCN=C(NCCCc1nccs1)N1CCC(C(O)C(F)(F)F)C1 48314,S(=O)(=O)(c1cc(-c2ccccc2)no1)C1(C(=O)O)CC1C(F)(F)F 48315,C#Cc1cccc(C(=O)NCC(C)(CC)NC(C2CCCCN2C)=O)c1C 48316,c1(C(=O)NCC(C)N(C(c2c(C)nns2)=O)C)cc(C2(Cl)CC2)n(C)n1 48317,C(=O)(C(C)(C)C(C)NC(=O)CCc1cn[nH]c1)NC(c1nccc(O)n1)C 48318,S(=O)(=O)(c1ccc2c(c1)nc(C1CCCCC1)n2CC)N(C(COCC)(C)C)C 48319,CC(C)CC(O)C(=O)N1CCN(C(=O)Cn2ccnn2)CC1c1cccc(F)c1 48320,CC(C)CC(C)(O)CNC(c1cc(CNC(C2(C)CC2C)=O)ccn1)=O 48321,c1(C(N2C(C(N(C)Cc3scc(C)n3)=O)C(C)CC2)=O)ncn2c1CCC2 48322,CCCC(CNC(c1coc(C(C)C)n1)=O)C(=O)Nc1cn(C)nc1O 48323,C1(CNC(COC(CC)(C)C)=O)C(C2CC2)CCN1C(c1cnc(C(F)F)s1)=O 48324,C1(C(N(CCNC(CCOCC)=O)C(C)C)=O)CCC(N2CCOCC2)CC1 48325,C=CCCCCCCCC(=O)N1CC2(CCCC(CNC(C3(O)CCC3)=O)O2)C1 48326,Cc1cc(Br)cnc1C(=O)NCC1CN(C(c2ccc(Cl)o2)=O)CC1C 48327,C(=O)(C1=NN2CCCN=C2N1)NC1C(NC(Cc2cc(C)sc2)=O)CCCC1 48328,c1(NC(C)=O)nc(C(=O)NCC(C)NC(C2CC23CC3)=O)cs1 48329,c1(C(=O)NC(CNC(c2cc(CC)c(CC)o2)=O)C(C)C)c(F)ccc(C)c1F 48330,N1(C(C2(CC(C)C)CCC2)=O)CC(NC(=O)Cc2coc(C(F)F)n2)C(C)C1 48331,C1(C)(C(=O)NCC(C)NC(c2cnn(-c3ccccn3)c2)=O)CC=CCO1 48332,N1(C(C(CCC)OC)=O)CC2CC(NC(=O)CC3(O)CCOCC3)CC1C2 48333,c1(C(N(C2CCN(C(c3ccc(CC)s3)=O)C2)CC)=O)c(OC)nsc1OC 48334,C1(OC(CCCOCC(C)C)=O)CCCC(C(C)(C)C)CC1 48335,C(C(=O)NCCC1CN(C(c2cnccc2Br)=O)C1)(C(C)(C)C)NC(C)=O 48336,N1(C(C(C)(CO)NC(C)=O)=O)CC(NC(c2ccn(CC(C)C)n2)=O)C2(CCC2)C1 48337,C(CO)(C(C)NC(=O)Cn1nnc(C2CC2)n1)NC(C=C(CC)C)=O 48338,C(C(C)C(C)C(=O)NCCOCCN(C)C(c1cc(C)nn1C)=O)OC 48339,C1(CC#C)CN(C(C2CCN2C(=O)COCC2CCCO2)=O)CCO1 48340,C1(Cl)(C(N2CCC(N(CCC)C(c3nocc3CC)=O)C2)=O)CC12CCC2 48341,N1(C(c2ccc(CC)cn2)=O)CC2CCCC(C1)N2C(c1oc(C)nc1C)=O 48342,c1(C(N2CC3(CN(C(c4cccc(C)c4)=O)C3)C2)=O)c(N)cc(Cl)nc1Cl 48343,C=CCC(CC=C)C(=O)NCC1CN(C(=O)CC2CCC(=O)NC2=O)CCN1C 48344,c1(C(=O)NCCC(CCC)C)ccc(C(C)(C)C)c(F)c1 48345,c1(-c2cn(CCNC(C34CC(CO3)C4)C)nn2)ccc(Cl)cc1OC(F)(F)F 48346,c1(NC(CC)CC(F)(F)F)ncccc1S(=O)(=O)NC(c1nncs1)C 48347,Cc1nccc2c(=O)c(-c3noc(C4CCC5(C=C5)OC4)n3)c[nH]c12 48348,c1(CNC(=O)CCNC(=O)CCCn2cncn2)cccc2cncn12 48349,c12nc(C)c(o1)C(=O)NC2.C(CCCCC1CC1)NC(CN(C(C)=O)C)=O 48350,C(N=c1[nH]c(=NC(C)CCC2CC2)c2c(ncn2C)[nH]1)c1cccc(C)c1N 48351,C1(C(=O)NC2CCN(CCC)C2)CN(C(c2cncs2)=O)CCO1 48352,Cc1cn2c(n1)CCC(C(=O)NC1CCC1NC(c1ccccc1[N+](=O)[O-])=O)C2 48353,C(=O)(C(CC(C)C)C(C)C)N1CC(CC=C)(NC(=O)COC2CCN(C)CC2)C1 48354,C(CCCC(=O)NC1CCOCC1C(=O)N(CC1=CCCOC1)C)(OC)OC 48355,c1(C(N(CCNC(=O)CCCn2ccnc2)CC)=O)c(F)ccc2cnn(C)c12 48356,C=C1CCC(NC(c2nc(C(=O)Nc3ccsc3COC)cs2)=O)CC1 48357,Cc1csc2c(C(N3CC4CC(NC(=O)Cn5cnnn5)CC3C4)=O)ncnc12 48358,C(=O)(C(O)CCC(F)(F)F)N1C(C(C)C)C(NC(C2CCSC2)=O)CC1 48359,C1(C(=O)NC2CC(CCNC(C3CCC(OC)CC3)=O)C2)CCc2nncn2C1 48360,c1(C(N2CCC(N(C(=O)CC(C)F)CC)CC2)=O)ccc(-n2cnnn2)c(C)c1 48361,C1(C(=O)NCCC2CN(C(C3(C)CCC3)=O)C2)CC12CCCCC2 48362,c1(C(=O)NC2C(NC(C(C)n3ccnn3)=O)CCC2)cccc(Cl)c1Cl 48363,C1(C(=O)NC(C(=O)NCCCN=[N+]=[N-])C2(C)CC2)CCCC(=O)C1 48364,N1(CC(COCC(C)C)O)CCC(N(C)C(c2cnon2)=O)CC1 48365,C(=O)(C1=CC2C=CC(C1)C2)NCc1c(C(N2CCC(N=[N+]=[N-])CC2)=O)nco1 48366,C(C1CCCC1)=C(C)C(=O)N(CC(O)C(=O)N1CC(c2noc(C)n2)C1)CCO 48367,N1(C(C(C)NC(CC)(C)C)=O)CC(C)C(NC(C2C3CC4C(C3)C24)=O)C(C)C1 48368,Cc1ccc(C)c(C(=O)NC2CN(C(=O)CCc3c(C)noc3C)CC2F)c1O 48369,c1(SC(c2cccc(Br)c2)C(=O)OC)c(C)nn(C)c1C 48370,c1(C(N(CC(C)NC(CC(C)(C)OC)=O)C)=O)nccc(Br)c1C 48371,CC1(CNC(C2CCCC3(CC3)C2)=O)CN(C(c2cn3ccnc3s2)=O)CCO1 48372,C1(NC(COC2(C)CCC2)=O)C2CCCN(C(=O)CN3CCNC3=O)C2C1(C)C 48373,c1(C(CNC(=O)NC(c2ccccc2)Cc2ncc[nH]2)F)ccc(Br)cc1 48374,C12(NC(C(C)=C(C)C)=O)COC(C1)C(NC(c1n[nH]cc1C(F)(F)F)=O)C2 48375,c1(CC(N2CC(CCC)N(C(=O)CN(C)CC)CC2)=O)ccc2c(c1)CCN2C 48376,N1(C(CC(CCC)O)=O)CC2CCC(C1)C2NC(c1cc(C)on1)=O 48377,c1(NC(c2c(C)nns2)=O)cnc(F)cc1C(=O)Nc1cccc(CCO)c1 48378,C1(NC(C2CCCC(O)C2)=O)CN(C(c2ccsc2C(F)(F)F)=O)CCC1CO 48379,Cc1ccc(F)cc1N(C)C(C1CCCN(C(c2ccn(C(C)C)n2)=O)C1)=O 48380,N1(C(CN(C(C)C)C)=O)CCCC(NC(c2cc(NC3CC3)ncc2Cl)=O)C1C 48381,C(=O)(CS(=O)(=O)CCC(F)(F)F)NCC1C(NC(C(C)O)=O)COC1 48382,C1(NC(C(C)OCCCCCC)=O)CN(C(=O)C(F)OC)CCC1(C)C 48383,CCC(C)(CNC(=O)C1=NOC(CNC(c2cc(C(N)=O)co2)=O)C1)C(N)=O 48384,S(=O)(=O)(c1cccs1)NC(C)C(=O)NCC(CO)NC(=O)Cn1cccnc1=O 48385,C1(NC(C=CC)=O)CCN(C(C2CC(=O)OC2(C)C)=O)C12CCC2 48386,c1(C(=O)NCCC2N(C(C3(OC(C)=O)CC3)=O)CCC2)cnc2onc(C)c2c1 48387,c1(C(=O)NCC2COCCN2C(=O)CC23CCCC2C3)nccc(Br)c1O 48388,C(=O)(C(C)CS(C)(=O)=O)N1C(CCOC)CN(C(=O)CCc2cnoc2)CC1 48389,c1(-c2nc(NC(CCC)=O)sc2)ccc(F)c(C)c1.c12ccsc1c2=O 48390,N(C1CCCc2c[nH]nc21)C(C(CC1CCC1)NC(c1cccc(OC)c1)=O)=O 48391,C1(CNC(C2CCCC(C)C2)=O)CC2(CC2)CN1C(C1CCCN1C)=O 48392,c1(N2CCC(C)(COC)C2)ccc(Br)c(S(=O)(=O)NCCC(C)CCO)n1 48393,N1(C(C2CC(OC)C2)=O)CCCC(C)(NC(=O)COCc2ccncc2)C1 48394,CS(=O)(=O)c1nc(Cl)cc(=NC2CCCCC2NC(C2CCCOCC2)=O)[nH]1 48395,CC(C)(C)C(CO)C(=O)NCC(F)CNC(=O)CCc1cccc(C(F)(F)F)c1 48396,C(=O)(C(F)C(F)(F)F)N(CCCN(C(C(N1C(C)CCC1C)C)=O)C)C 48397,c1(C(N(C)CCNC(=O)CCc2ccc(CO)cc2)=O)sccc1S(C)(=O)=O 48398,C1(NC(c2nncs2)=O)CC(O)(C2CCN(C(c3ccccc3)=O)CC2)C1 48399,CCCC(CC)C(=O)N(C(C)(C(=O)Nc1ccc(O)nc1)C1CC1)C 48400,c1(NC(CNC(C2C(c3ccccc3)(C)C2)=O)C2CC2)ccn2nccc2n1 48401,N1(Cc2scc(C)n2)CCC2(CC1)CN(C(C1(C)CCOC(C)C1)=O)CC(C)O2 48402,C1(C(N2CCCC(C)C2)=O)CCN(C(=O)CCCC2CCC2)C12CCC2 48403,N1(C(CC(CC)O)=O)CCCC(C2CC2NC(c2cc(C)nn2CC)=O)C1 48404,N1(C(C2CCCCC(=O)N2)=O)CCCC12CCN(C(C1CC1F)=O)CC2 48405,C1(C(=O)NC2CCN(C(CC3(C#N)CCC3)=O)CC2)CCc2ncccc2C1 48406,C(CC(O)C(=O)NC(C1CCN(C(=O)COC2CCN(C)CC2)C1)(C)C)SC 48407,C(=O)(C(O)C(C)(C)C)N1CCN(C(CNC(C(C2CCC2)OCC)=O)C)CC1 48408,c1(NC(Cc2cccc(-c3ccc(OC)c(OC)c3)n2)=O)c(Cl)nc(C)nc1Cl 48409,C1(C(N2CCC(CN=[N+]=[N-])C2)=O)CCOCC1NC(c1cnsc1)=O 48410,CC(C)(C)CC(O)CC(=O)N1CCCN(C(c2noc3c2COCC3)=O)CC1 48411,C1(C(N2CC(CC(=O)OCC)C2)=O)CN(C)CCN1C(=O)CCc1ccco1 48412,c1(OCC)cc(NC(=O)C(N2CCOC(CC)C2)=O)cc(C)c1 48413,C(=O)(CCC(C)NC(C1CN(C(=O)C(C)c2cc[nH]n2)CC1C)=O)OC 48414,C(=O)(C(COC)COC)NC(CC(=O)NC(COC)COC)C1CC1 48415,c1(OC)cc([N+](=O)[O-])ccc1OCCNCc1ccc(OCC2CC2)nn1 48416,N1(C(=O)OC(C)(C)C)CCOC(CCSc2cnoc2-c2ccc(Cl)s2)C1 48417,C1(NC(CN(CCC)C)=O)CCN(C(c2cccc(N)c2C)=O)CC1O 48418,CN1CC=C(CC(=O)N2CCC3CCN(C(=O)CN4CCCNC4=O)C3C2)CC1 48419,c1(OC)nc(N2CCN(C(c3cc(Cl)c(Cl)s3)=O)CC2C)ncc1Br 48420,C1(CNC(c2ncc(C)cc2C)=O)CC2CCCC2N1C(c1cc(Cl)n(C)n1)=O 48421,N1(C(C(CSC)OC)=O)CCC(C2CCN(C(c3cnc(C(C)C)s3)=O)CC2)C1 48422,C(=O)(CC(O)CN(C)C)N(CCN(C(CCn1c(C)ncc1)=O)C)C 48423,C(CC(N)=O)(c1cn(CCS(=O)(=O)N(C)C)nn1)NC(CSC)=O 48424,N1(C(C(CCOC)C)=O)CCC(C(N2CCC(C)(CN(C)C)C2)=O)C12CCC2 48425,C1(COC)(NC(=O)CNC(c2cccs2)=O)CN(C(c2cocn2)=O)C1 48426,NC1(C2CCN(C3(C(=O)NC4CCCCC4)CC3)CC2)CC1 48427,C(=O)(CCS(=O)(=O)NCC1(O)CCN(C(=O)Cc2ccccc2C)C1)OC 48428,C1(NC(c2nccs2)=O)CCCCC1C(=O)Nc1ncccc1-c1ccccc1 48429,c1(C(=O)NCC2CC(F)(CNC(Cn3c(C)ccn3)=O)C2)ccnc(CO)c1 48430,C1(C(=O)NC2CC(CNC(c3c(C)nsc3NC)=O)C2)Cc2cc(F)cc(F)c2O1 48431,C(CC(C)C)(CS(C)(=O)=O)NC(c1cn(CCC)nc1C)c1nnnn1C1CC1 48432,C1(NC(=O)CC2CCC2C2CC2)CCCCN(C(=O)CC(F)(F)Cl)C1 48433,Cc1ccc2c(N3CCC(O)C3C(N3CCNCC34CCC4)=O)ncnc2c1 48434,C12(C(=O)NC(CC)CNC(=O)COc3cccc(Cl)c3)CCC(COC)(CC1)C2 48435,c1(C(=O)NC2(CN(C)C(c3sccc3-n3cnnn3)=O)CC2)cc(=O)n(C)cn1 48436,c1(C(C)C)c(C(F)(F)F)n[nH]c1C(=O)NCC=CCNC(C1CCC(=O)O1)=O 48437,C1(C(=O)NCC=CCNC(CSCCN(CC)CC)=O)CCCCC1CC 48438,N1(C(C(Cn2ccc(C)n2)C)=O)CCCC12CCCN(C(=O)C(C)CC(C)C)C2 48439,C12(C(=O)NC(c3cnc(C)s3)C)C(NC(=O)Cn3cnnn3)C3CC1C2C3 48440,c1(C(=O)NCC2(O)CCCN(C(COC(CC)(C)C)=O)C2)ccc(C#N)c(O)c1 48441,C=CC(C)(C)C(=O)N(CCCNC(=O)C(N1CCCC(O)C1)C)C 48442,Cc1nc2ccccc2cc1C(=O)N(C)CC1CC(F)CN1C(=O)C(C)O 48443,CN1CCCC(CNC(=O)C(O)CNC(c2ccccc2F)=O)C1 48444,c1(CC)ccc(NC(C2(N(C)C(C3(CC)COC3)=O)CC2)=O)cc1O 48445,C1(C)(CNC(C(C)N2CCC2)=O)CN(C(c2ccc(F)c(Cl)c2F)=O)C(C)(C)C1 48446,Cc1cc(C(=O)N(C(C)(C(=O)N2CC(OC(=N)O)C2)C2CC2)C)nn1C 48447,n1(CC(=O)N(CCOC)CCNC(=O)C(C2CCC(=O)N2)C)nc(C)c(Cl)c1C 48448,C1(C(N(CC(C2CCC2)OC)C)=O)CCCCC1(C)NC(c1cnc[nH]c1=N)=O 48449,N1(C(C(c2cccs2)SC)=O)CC2(C1)CN(C(c1ccc(Cl)cc1F)=O)C2 48450,C12(COC)CC(CN1CC1C(O)CCN1C(=O)OCc1ccccc1)C2 48451,C=C(C)C1OCCCC1C(=O)NC1CN(C(c2ccccc2C(C)C)=O)CC1O 48452,N1(C(CC2C(C)CCCC2)=O)CCC=C(C(=O)NCCN(C)C2CC2)C1 48453,Cc1ccc(F)c(O)c1C(N1CC(CNC(=O)CCc2ccon2)C(C)C1)=O 48454,C1(n2cc(CC(C)(C)O)nn2)CCCCCN1C(=O)CCC12CCC(CC1)C2 48455,c1(C(C(=O)NCCCOC)N(C2CN3CCC2CC3)C)ccc(F)c(Br)n1 48456,C1(CNC(C(C)N(C(=O)C(C)O)CC)=O)NC(=O)NC1=O 48457,CC1=C(C(=O)NC2CCOCC2NC(C2CC(CN(C)C)C2)=O)CCS1(=O)=O 48458,C12(C(=O)NCCNC(CO)C(F)(F)F)CCCN1CC(O)C2 48459,CCC(C)C(=O)C(=O)N1CCC(C)(C(=O)NCC2CCCC2)C1 48460,c1(C(=O)NC2C(C)(C)CN(C(C3(C)CCNC3=O)=O)C2)c(F)ccc2occc12 48461,C(C(C)(CC(C)C)NC(=O)C(C)N(C)C)NC(C1(CC)CC1)=O 48462,Cc1c(C(=O)NC2CC2NC(c2ccc(C(F)(F)F)o2)=O)cnn1C1CC1 48463,N1(Cc2n(C)cc(C(=O)O)c2)CCC(O)C(C(=O)O)(N(C)C)C1 48464,c1(C(N2CCC(OC)(CNC(C3(C)CCSCC3)=O)C2)=O)ccc(=O)n(C)c1 48465,C=C(CNC(C1C(O)CCN1C(c1cccc2occc12)=O)=O)C1CCOCC1 48466,C12(NC(=O)COC3CC3)CCC(C(=O)NCC(O)C3CCC3)(CC1)C2 48467,N1(C(c2cnn(CC(F)F)c2)=O)CCC12CN(C(C13CCCCC1C3)=O)C2 48468,N1(C(c2n(C)ccn2)=O)CCC(C2CCN(C(c3cnco3)=O)CC2)C1 48469,N1(C(C2CC(C)(c3ccccc3)C2)=O)CCCCC12CC2 48470,C1(C(=O)NC(C2CCCC2)C#C)CCC2(CC2)N1C(=O)CC1(OC)CCC1 48471,N1(C(Cn2ncc(C)c2)=O)CCC2(CC1)CC2NC(C12CCC1C2)=O 48472,c1(N2CCC(CCN(C)CC)CC2)nccc(N(C)CCN2CCCC(O)C2)n1 48473,c1(OCC)cccc(NC(=O)C=CC(N2CCCCC2CNC(=O)CC)=O)c1 48474,c1(C(C(=O)NC2CCC(N(C(=O)C(C)(C)CF)C)C2)=O)c[nH]c2cc(F)ccc12 48475,CN=c1nc(C(N2CC(NC(=O)C(C)(C)C(F)(F)F)CC(O)C2)=O)cc(C)[nH]1 48476,N1(C(C2CC(=C)C2)=O)CCC2OCCN(C(=O)CCc3ccc(SC)cc3)C2C1 48477,N1(C(CC=CC)=O)CCCC2(CCC2NC(C2CCCCO2)=O)C1 48478,n1(CCC(=O)NCCC(C)NC(c2c(C(=O)OC)scc2)=O)c(C)csc1=O 48479,c1(C(N2CC(C)C(CCNC(c3cccc(F)c3)=O)C2)=O)cncc([N+](=O)[O-])c1 48480,C1(NC(c2cc(SC)oc2)=O)CC(NC(=O)C2=CCCOC2)C12CCOCC2 48481,N1(C(=O)OC)CC2CCC1C(C(=O)NCCCCNC(C1(CSC)CCC1)=O)C2 48482,C1(CNC(CC(C)OC)=O)CCN(C(=O)Cc2ccccc2)C12CC2 48483,C1(c2n(C(C)C)nnn2)(NC(CC(N)=O)C2CCOCC2)CCOCC1 48484,C(=O)(C(Cc1ccoc1)NC(=O)C(F)=CC1CC1)N(CC(C)OC)C 48485,c1(CC)nnc(N2CC3(CN(C(=O)CCCn4cccn4)C3)C2)c(C#N)c1CC 48486,C1(CNC(c2c(C)ocn2)=O)CC2CCC(C1)N2C(=O)CS(=O)(=O)N(C)C 48487,CC1(CNC(=O)Cn2ccc([N+](=O)[O-])n2)CN(C(c2cccnn2)=O)CCO1 48488,C1(NC(CCc2cccc(OC)c2)=O)CN(C(c2ccc[nH]2)=O)CCCO1 48489,c1(C(=O)NCC(CC2CN(C(CCCCC)=O)C2)(C)C)ccc2oncc2c1 48490,c1(C(=O)NC2C(NC(C3(COC)CCCCO3)=O)CC2)cc(C)ccc1C 48491,N1(C(c2nnn(CC)c2C)=O)CCC(NC(C2(Cl)CC2(C)C)=O)CC(O)C1 48492,C1(NC(c2cnc(CCCC)s2)=O)CN(C(C2(CC)CCNC2=O)=O)CC1C 48493,N1(C(CCC2(NC(C3(C)CCC(=O)N3)=O)CCC2)=O)CC2CCC2(C)C1 48494,C1(C(=O)NC2C(C)N(C(C3COC(C)(C)CO3)=O)CCC2)CCC(C2CC2)CC1 48495,S(=O)(=O)(c1ccc(NCC2CCOC2)c(C#N)c1)N1C(C)CN(C)CCC1 48496,CC1CSCCN(C(=O)CC2CCCC(NC(=O)C(c3ccnn3C)O)C2)C1 48497,C1(NC(Cn2cc(CNC(C3CC(C)OC3)=O)nn2)=O)CC(C)(C)C12CCC2 48498,C1(C(N2CC(CNC(Cc3cn(C)nc3)=O)OCC2)=O)CC2C=CC1C21CC1 48499,c1(OC)cc(C(=O)NC2CN(C(c3ccoc3Cl)=O)CC2F)cc2nc(O)[nH]c12 48500,c1(C(=O)NC2CC3(C(NC(CC4N(CC)CCC4)=O)C3)C2)ccn2c1CSCC2 48501,c1(NC(C2NCCN(C(c3nc(CC)oc3)=O)C2)=O)cc(C)cc(Br)c1F 48502,Nc1ccc(C(=O)NC2CCCN(C(c3cncc(F)c3Cl)=O)CC2)nc1Cl 48503,C=Cc1cnn(C)c1C(N1CCN(C(=O)CC2(C)CC2(Cl)Cl)C(C)C1)=O 48504,N1(C(Cc2cccc(COC)c2)=O)CCN(C(=O)CCCCSC)C2COCC12 48505,N1(C(C2CC(C(=O)O)CN(C(=O)OC(C)(C)C)C2)=O)CCC(NC(C)C)C(O)C1 48506,CC1CN(C(c2ncn3c2CCC3)=O)CCCN1C(c1cccc(N)c1)=O 48507,N1(C(C2OCCN(C(C)C)C2)=O)CCN(C(=O)Cc2sc(O)nc2O)CCC1C 48508,C(=O)(C1=C(Cl)CCCC1)N1C(C)CC1C(=O)NC1(CO)CCCCC1 48509,CCCC(C)CC(=O)N1CCCCC(NC(c2cc(C)c(C(=O)OC)o2)=O)C1 48510,N1(C(c2ccc(CN(C)C)cc2)=O)CCC=C(CNC(=O)CC2CCC3CC23)C1 48511,c1(N2CCCC(C(C)NC(C(Br)=C(C)C)=O)C2)nc(N(C)C)cc(C(F)(F)F)n1 48512,c1(C(=O)NCc2nc(CNC(CCc3nc(=N)[nH][nH]3)=O)sc2)cccnc1S 48513,N1(C(C2N(C(Cn3nc(C)oc3=O)=O)CCC2(C)C)=O)CCC2(CCCCO2)C1 48514,Cn1nnc2c(C(N3CCC(N(CCO)C(C4CCC(F)CC4)=O)C3)=O)ccnc12 48515,c1(C(=O)NC2CN(C(C(C)OCCOC)=O)CC2C)c(C)cccc1Br 48516,N1(C(C(OCC)OCC)=O)CCC(F)(C(=O)NCC(C)(C)CN2CCCC2)CC1 48517,Cn1nc(Br)cc1NC(C1CCCN1C(=O)COc1ccccc1)=O 48518,C(N=c1[nH]c2ncc(Cl)cc2o1)c1c(C)c(C(F)(F)F)n[nH]1 48519,c1(C(=O)NCCC(C)NC(C2C3CCCCCC23)=O)c(F)ccc(F)c1Cl 48520,Cc1ccc(CCCC(=O)NC(C)(CNC(C2CCCCC2O)=O)C2CC2)cc1 48521,C1(C)(C(N(C2CCN(C(=O)CCC3CCC(C(N)=O)O3)CC2)C)=O)CCC(=O)N1 48522,c1(C(=O)NCCCN(CCOCCOC)C)cc(C)nc2c1nc(C)n2C 48523,c1(C(=O)NC2CC(NC(C(Cn3ccc(C)n3)C)=O)C2)nccc(F)c1Cl 48524,C1(N(C(C2C(CCC)CCC2)=O)C)(N(C)C)CCCCC1 48525,C1(C(N2C(CCCNC(CCC=C)=O)CCC2)=O)CCOC(C)(C)C1 48526,Cc1cc(C(N2CC(C(C)NC(c3cc4occc4s3)=O)C2)=O)cc(N)c1O 48527,C1(COC)(NC(c2cc[nH]c(=N)c2)=O)CCN(C(=O)C(C2CCOCC2)C)CC1 48528,C1(NC(CCOCC(C)C)=O)CCC2CCN(C(c3c[nH]ccc3=O)=O)C12 48529,c1(C(c2nnnn2C2COC2)NCC(C2CCSCC2)(C)O)cccc(CO)c1 48530,N1(C(C2(C(=O)OC)CC(=C)C2)=O)CC2CCC1CN2C(C1CCCO1)=O 48531,CC1(C#CC(=O)N2CCCC2(C)CNC(=O)C(C)(C)C2CC2)COC1 48532,C12(C(N3C(CCNC(c4cnc(COC)s4)=O)COCC3)=O)CCCC1OCC2 48533,C1(CS(N)(=O)=O)CCCN(C(=O)CNC(C2CCNCC2)=O)C1 48534,N1(C(c2cccs2)=O)CC(CNC(C2(C(F)(F)F)CCC2)=O)CC12CCOCC2 48535,c1(C(=O)NCCCN(C(=O)CN2CCC(C)C2)CC)sc2cc(F)ccc2c1C 48536,c1(CC(=O)NC(C(C)NC(=O)Cn2cnnn2)CO)coc2ccc(F)cc12 48537,c1(C(=O)NCC2(O)CCCN(C(c3cc(Cl)no3)=O)C2)ccc2c(c1)CCCO2 48538,N1(C(C2CCN2C(c2cccnc2C(F)F)=O)=O)CC(Sc2ccccc2)C(F)C1 48539,CCCCCC(C)(C)C(=O)N1CC(CO)(NC(c2c[nH]c3cccc(F)c23)=O)C1 48540,CC1CN(C(=O)OC(C)(C)C)CCS1(=O)=O.C12(F)CN(C1)C(=O)N2 48541,c1(OC)ccccc1OC1CCN(C(=O)C(=O)NCC2(C)COC(=O)N2)C1 48542,C(=O)(CCCCCC(C)C)N1C(C)CCC(NC(C2(CC=C)CC=CC2)=O)C1 48543,N1(C(CCN(C(CCC2C(C)(C)C2)=O)CCO)=O)CCc2nc[nH]c2C1 48544,C(c1ccc(C)c(C)c1)=CC(=O)NC1C2(CC(NC(C(CC3CC3)OC)=O)C2)C1 48545,Cc1cc(C(=O)NC2CCC(NC(C3CCC(C)CC3)=O)C2)sc1C 48546,Cc1ccc(C(N2CCN(C(c3ccc(O)cc3)=O)C(C3CC3)C2)=O)nc1O 48547,Cn1ncc2c1CCCC2N=c1[nH]c(=NCC2SCCS2)[nH]c2cc[nH]c12 48548,C1(CCO)CCN(C(=O)NC2(CNC(=O)OC(C)(C)C)CCCCC2)CC1(C)C 48549,c1(N2CCN(CC)CC2)nc2cccnc2c(=NCC2CCCC(F)(F)CC2)[nH]1 48550,c1(C(=O)Nc2cccc(NC(CC3C(CC)C3)=O)c2)c(Br)c(C)nn1C 48551,C1(F)(C(N2CCC(NC(Cc3c(C)con3)=O)CC2)=O)CS(=O)(=O)CC12CCC2 48552,C(=O)(C#CC1CCCOC1)NC(C1CCCN1c1ncnc2[nH]cnc12)(C)C 48553,Cc1cc(F)sc1C(=O)NC1CCC(CNC(c2ccc(-c3cc[nH]n3)s2)=O)C1 48554,C1(NC(=O)CSC2CC2)CN(C(=O)C(O)CC2CCOCC2)Cc2ccnn2C1 48555,c1(OC)ccc2c(c1)N(C(c1ccc(Br)cc1Cl)C(=O)NCC(F)F)CCC2C 48556,c1(C(c2n(CCOCC)nnn2)N)cnc2c(c1)CCC2.C(CCO)CC1CCC1 48557,c1(C(=O)OCC)ccc(CCNC(=O)C(=O)NC(C)C(C)(C)C#N)cc1 48558,N1(S(CC)(=O)=O)CCCC1C(N1CCC1CNC(=O)CCNC(=O)COC)=O 48559,CCCCCCC(=O)N(CCCNC(c1sccc1C(F)F)=O)CC 48560,C1(NC(CC2C(C#N)C2)=O)C2CN(C(c3cnn(-c4cccnc4)c3)=O)CC12 48561,Cc1cc(C(N2CCCC(NC(C3C=CCC3)=O)C2C)=O)c(O)c(C)n1 48562,c1(OC)cccc(C)c1C(N1CC2CC1(CNC(=O)CN1CC3CCC1C3)C2)=O 48563,N1(C(c2c(C)n[nH]c2)=O)CCCC2(CCC(NC(=O)C(=O)N(C)C)C2)C1 48564,N1(c2cc(C(C)=O)ncn2)CCN(C(c2cc(C)c(C)nn2)=O)CCC1C 48565,n1(CC(=O)NCC2CC(NC(=O)CCc3cnoc3)C2)ccccc1=O 48566,C(C)(C(C(=O)N1C(CO)CC1C)C(C)C)NC(C1ON=C(CC)C1)=O 48567,CCC(COC)(CC)C(=O)N1CC(CCNC(=O)CO)(OC)C1 48568,c1(C(N(CCC)CCNC(C2CC=CC2)=O)=O)ccnc(-n2cccc2)c1 48569,c1(NC(c2c(NC(C(CCC)C)=O)ccs2)=O)ccc(Cl)cc1Br 48570,c1(C(=O)NC2CC(CNC(C(n3ncc(C)c3)C)=O)C2)ccc2cccnc2c1 48571,CC1CN(C(c2nnn(C)c2C(F)F)=O)CCC1N(C)C(c1cc(Cl)n(C)n1)=O 48572,C#CC1(O)CCN(C(C2CCCC(NC(=O)CNC(=O)NC)C2)=O)C1 48573,C1(CCC=C)CCCN(C(C23CC2CCN3C(=O)C(=O)NOC)=O)C1 48574,CC1CN(C(c2cncn(C)c2=O)=O)CCC1N(C)C(c1ccc(CO)cn1)=O 48575,CC(C(C(=O)O)NC(C1CCCN1C(=O)OC(N)=O)=O)OC(C)(C)C 48576,C=CCC(CC)C(=O)N1CC2(CC(CC(N3CCC(c4ccon4)C3)=O)C2)C1 48577,c1(N2CC(C)N(C(=O)CN(C)C)CCC2)ncnc2c1c(Br)cn2C 48578,C12(C(N(CC(=O)N(C)CCc3cnccn3)C3CC3)=O)CCCC1C2(F)F 48579,c1(C(C(=O)NCC(CNC(CSCCN(C)C)=O)(C)O)O)cccc([N+](=O)[O-])c1 48580,CC1CCCC(CCNCC(C(=O)OCc2ccccc2)C)C1 48581,c1(CCN(C)C(=O)NC23CCC2C3)ccc(NS(C)(=O)=O)cc1.C1CCC(=O)N1 48582,c1(C(=O)OC)cn(C)[nH]c1=NC(=O)C(c1ccccc1)OC(c1ccccc1)=O 48583,c1(C(N2CC(NC(CN(C3CC3)CC)=O)C(C)C2)=O)c(C(F)F)nn(C)c1C 48584,N1(C(COC)=O)CC(CNC(c2c(F)ccc(Br)c2Cl)=O)C2(CCC2)C1 48585,c1(C(N(CCNC(C2C(CC)C2)=O)CC)=O)cnc(C(F)(F)F)c(F)c1 48586,C(=O)(C1=CCN(C(C2CCNC(=O)C2)=O)CC1)NCC(C)(C1CC1)OC 48587,C(CCCCC(=O)NCC1C(C)CCN1C(=O)CC1(C)CC1(Cl)Cl)OCC 48588,C(=O)(CC(CC)SC)N(CCC)CCNC(=O)COCCF 48589,C1(CNC(C(CC)N(C)C)=O)(NC(C23CC(C(=O)N(C)C)(C2)C3)=O)CC(F)(F)C1 48590,CCC(CCOC)C(=O)N1CC(CNC(c2cc(=O)cc(Cl)[nH]2)=O)C2(CC2)C1 48591,N1(c2cc(C(=O)OC)nc(Cl)n2)CC2(C1)SCCC2NC(=O)Cc1n[nH]c(C)n1 48592,c1(NC(=O)NC2(C(=O)OC)CC2)ccc(NC2(C)CCC2)c(OC)c1 48593,C1(C)(CC)COCCC1C(=O)NC1(C(=O)N2CCCCO2)CCCC1 48594,N1(C(C(COC)OC)=O)CC2CCC(NC(=O)CCS(C)(=O)=O)C2C1 48595,c1(C(N2CCOCC(O)C2)=O)cccc2c1CCN(c1ncnc3[nH]ccc13)C2 48596,c1(COC)c(C(=O)NC2CCN(C(c3ccc(NC4CC4)nc3)=O)C2C)cnn1C 48597,Cc1cc(=NC(C)CCCC(F)(F)F)[nH]c(=NCC2CC23CCC(O)CC3)[nH]1 48598,C1(C(=O)NCC(C(C)C)CO)C2CC3C(C2NC(c2ccccn2)=O)C13 48599,c1(C(=O)NC2CN(C(c3cc(C)ns3)=O)CC(C)(C)C2)cnc2ncnn2c1C 48600,c1(CC(=O)NC2C(C)CN(C(=O)CCCCN(C)C)C2)ncn2c1CCC2 48601,CCC(C)(C(=O)N1CCC(CCNC(=O)C(O)Cc2cnc[nH]2)C1)OC 48602,C1(c2ccc(CC)o2)CCCCCN1N1CCOCC1CC 48603,O=C(CCCC(F)F)NCC1CCN1C(c1ccc(CO)nc1)=O 48604,C1(=CCNC(c2ccc(SC(F)(F)F)cc2)=O)CCN(C(=O)C(O)CF)CC1 48605,Cc1ccc(C)c(NC(=O)C(C)N(C)C2CC2)c1.C12CCCN1C(=O)CC(=O)N2 48606,N1(Cc2ccccc2)CCN(CCc2nnnn2CC2CC2)CC1.c1ccccc1 48607,C1(C(=O)NC(c2ccccn2)(C)C)CCCCC1NC(C1CNC(=O)C1)=O 48608,c1(SC)ccnc2nc(=NC(=O)c3n[nH]cc3CNCC3COC3)[nH]n12.C(C)(C)C 48609,N1(C(CCC(C)C)=O)CCC2(CC1)CC(C)N(C(=O)CN1CCOCC1)C2 48610,C(=O)(C(C)CC(C)CC(C)C)NCC1(C)C(C)CN(C(C(C(CC)(C)C)O)=O)C1 48611,CCC(CC(=O)NC1CC(NC(c2cc(OC)cnn2)=O)C(O)C1)C(C)C 48612,CC(C(=O)OC(C)(C)C)C(=O)N1CC=CC1CNC(=O)C=Cc1nccs1 48613,C1(C(=O)NC2(CC=C)CN(C(=O)C(C)C)C2)C2CC2C2CC12 48614,Cc1noc(C)c1CC(C)C(=O)NCC1CCN(C(=O)CCc2cccnc2)C1 48615,C(C1CSc2ccccc21)NC(C(n1cc(CNC(CC)=O)nn1)C)=O 48616,c1(C(=O)NC2C3(NC(c4nc(C)[nH]n4)=O)CCC(C2)C3)cc(F)cc([N+](=O)[O-])c1 48617,C(C)(CN=c1ccnc(N2CCOC(C3CC(c4ccccc4)C3)C2)[nH]1)SC 48618,C=CCC(CNC(=O)CCc1ccccc1)C(=O)NCc1cc(C)cc(C)c1 48619,c1(CN2CCCC(NC(CCC(C)C)=O)CC2)cc(Cl)c(O)cc1F 48620,Cc1cc(F)ccc1C(=O)N(CC(C)C(=O)N(C)Cc1cccc(F)c1)C 48621,c1(C(N(CCC(C)NC(C2(OCC)CCOCC2)=O)C)=O)cc(F)c(Cl)cc1F 48622,Cc1cc(C(F)(F)F)sc1C(N1CC(C)C(F)C1)C(=O)NC1CCC1 48623,Cc1cc(=NCCN(C)C(C2Cc3cccc(C)c3O2)=O)[nH]c(C)n1 48624,C1(CC(=O)NCC(C)(C)CC2CN(C(c3ccncn3)=O)C2)CCC=CCC1 48625,Cc1ccc(-c2ccc(C(N3CCC(O)(C(F)F)C3)=O)cc2)cc1Br 48626,C1(NC(c2ccc(C#C)cc2)=O)CN(C(c2ccc[nH]2)=O)CC12CCC2 48627,N1(CCCC)CCC(O)C(C(=O)NC(c2ccc(OC)cc2)CC)C1 48628,Cc1ccc(C)c(CNc2cc(C(C)(C)C)cnc2Cl)n1 48629,N(C(=NCC1CN(C)S(=O)(=O)c2ccccc21)N1CCCC2(CC2)C1)C(CC)C 48630,c1(CNC(CCOCCN(C)C)=O)cn(C2CN(C(c3nocc3Cl)=O)C2)nn1 48631,N1(C(c2sncc2Br)C(=O)NCCCCCC)CCCC(NC(=O)OC)C1 48632,CC1CCC=C1C(=O)N1CCC(CO)(NC(c2cncc(C(F)(F)F)n2)=O)C1 48633,N1(C(C=CC)=O)CCC(C2CCCN(C(=O)CS(=O)(=O)CC(F)(F)F)C2)C1 48634,CC(C)CCCCCC(=O)N1CCC2CCCC12CNC(c1ncc(F)cn1)=O 48635,c1(C(N2CC(O)CC(NC(c3cc(C)[nH]n3)=O)C2)=O)csc2cc(Cl)cnc12 48636,CCC(CC)(C(=O)NCC1(C)CCN(C(c2ccc(CO)c(Cl)c2)=O)C1)OC 48637,N1(C(c2cn(CC)nc2C)=O)CCN(C(c2ccc(N)c(C)c2F)=O)C(C)C1C 48638,CC#CCC(C(=O)NCC1(C(=O)OC)CC1)NC(c1ccc(C)cn1)=O 48639,CS(=O)(=O)CCC(=O)NC(C(=O)NOC(c1ccccc1)C1CC1)C1CCCO1 48640,c1(OC)cnc(Cl)cc1C(N1CCC(NC(=O)C(C)(Cl)Cl)C(C)C1)=O 48641,C1(C(C)(C)C)(CNC(C(C)OCC)=O)CCN(C(C2CCC(N(C)C)CC2)=O)C1 48642,C(=O)(C1=NOC2(CCC2)C1)N1CC(C)N(C(=O)CCP(C)(C)=O)CCC1 48643,c1(C(=O)NC2C(OCC)CCCC2)n[nH]c2cc(C(=O)N=c3cco[nH]3)ccc12 48644,C1(CNC(CC2CCN(C)C2=O)=O)CN(C(c2cnc(S)[nH]2)=O)CC12CC2 48645,C(=O)(C1(C)CCn2ccnc21)NC(C(C)C)CCN(C)C(C1CSCCS1)=O 48646,C(=O)(CCC(=O)NN(C)C)NC(CC#CC)C(=O)NCc1oc(C)nc1C 48647,N1(C(C(=O)NCCCCCCCCCCCC)=O)Cc2ccccc2CC1(C)C 48648,CC1(C)CC(CNCCc2c(F)cccc2F)CCO1 48649,Cc1ccc(C(N2CCCC(NC(=O)C=CC(=O)OC(C)(C)C)C2CO)=O)c(Cl)c1 48650,C(CCCN=c1[nH]nc(C2CCCC2)s1)NC(c1cnn(CC2CCCO2)c1)=O 48651,N1(C(c2c(C)sc(-c3ccccc3)n2)=O)CC(F)(C(=O)O)C2(COC2)C1 48652,C1(NC(C2N(C(CC=C=C)=O)CC(O)C2)=O)CNC(=O)C12CC2 48653,CCC(CC(=O)NCC(C(C)C)NC(c1cccc(O)c1F)=O)C(F)F 48654,c1(CN2CCCN(CC(N)=O)CC2)cccc2c3c([nH]c12)CCCCC3 48655,N1(C(C(C(C)NC(C(C(C)C)C2CCC2)=O)C)=O)CC(=O)NCC12CC2 48656,S(=O)(=O)(c1ccc(Cl)nc1)NCC(C)NC(C1COC2(CCNCC2)C1)=O 48657,Cc1n[nH]cc1C(=O)NCCCOCCN(C(=O)COC1CC1)C 48658,n1(CC)ncc(C(N2CC(NC(=O)C(C)c3ccsc3)C2)=O)c1C(F)(F)F 48659,CC1=C(C)CC(C)(C(=O)NC2C=CCN(C(c3ncsc3S(N)(=O)=O)=O)C2)CC1 48660,C=CCCCCC(=O)NCC1CCC(Cn2cc(C(N)=O)nn2)CC1 48661,CC(CC1=CCCCC1)NC(=O)CCN(C(=O)C(O)CCN(C)C)CCO 48662,N1(C(c2cc(C)no2)=O)CCC(C)C(CNC(=O)CCCOC(C)(C)C)C1 48663,C1(C(N2CC(C3CN(C(CNC(C)=O)=O)C3)C2)=O)Cc2cccc(Cl)c2C(=O)O1 48664,C(=O)(CCCCC(N)=O)NC1CC(NC(C(CC(C)C)NC(C)=O)=O)C1 48665,Cc1ccc(NC(=O)C(C2CC=CCC2)NC(c2snnc2C)=O)cn1 48666,Cc1cccc(C)c1OCC(=O)NC1CCN(C(=O)CC2CCC2)C1C(C)(C)C 48667,C1(CC(=O)NC2CCC(NC(c3snc(O)c3Cl)=O)C2)SC2=NCCN2C1=O 48668,c1(CC(N2C3(CN(C(c4c(C)nns4)=O)C3)CC2)=O)n[nH]c2ccccc12 48669,c1(C(C)N(C)C(C2CCN(c3ccccc3Br)C2=O)=O)ccc(Cl)cc1 48670,C(CCCC(=O)N1CCC1C1CCCC1)NC(Cn1c(C)ccn1)=O 48671,c1(C(N2CC(CNC(C3CC3(F)F)=O)C(F)(F)C2)=O)ccc2cnoc2c1 48672,C1(NC(=O)C2=NOCC2)CC2(CCN(C(C3CCCCC34CC4(F)F)=O)CC2)C1 48673,CC1COCCC1N(C(=O)C(C1CCCO1)NC(=O)CCC1CCC(=O)C1)C 48674,N1(C(CCC(OC)OC(CNCC)(C)C)=O)CCCCC(C2CN(C(C)C)C2)C1 48675,C=CCC(C(=O)NC(CC(N)=O)C(=O)N1CCCC(C#N)C1)C(C)C 48676,N1(C(C2(C(C)=O)CC2)=O)CCC(C2CCN(C(c3ccc(Cl)s3)=O)CC2)C1 48677,c1(NC(C(COC(C)C)NC(C(CC)OC)=O)=O)ccc(OC(C)C)c(C)c1 48678,c1(OC)cnc(C(N2CC3C(NC(=O)Cc4c(C)noc4C)C3C2)=O)nc1 48679,N1(C(CC(C)(F)F)=O)CC2COCCC2(NC(c2ccnc3[nH]cnc23)=O)C1 48680,c1(C(=O)NC(C(C)NC(C23CC(O)C2C3)=O)C)ccc(Cl)cc1 48681,C1(NC(CC(COC)(C)O)=O)C2CC(O)C1N(C(=O)CCCc1cccs1)C2 48682,N1(C(c2ccc(CSCC)cc2)=O)CCN(C)C(CNC(=O)C(C)CCO)C1 48683,n1(CCC(=O)N(C(C2CCCCC2)CC2CCCC2)C)ncn(C)c1=O 48684,N1(C(C=C(C)C(C)(C)C)=O)CC2CCC2(CCNC(=O)C=Cc2cccn2C)C1 48685,C(=O)(C(C(F)(F)F)=Cc1ccccc1)N1C(CNC(c2c(C)csc2)=O)CCC1 48686,n1(CC(=C)C)nnnc1C(c1nc(C2CC2)cs1)NC(C1CCC1)C1CC1 48687,C1(C2CCC2)(C(=O)NCCCC2(NC(=O)CC3CCCC(=O)N3)CC2)CC1(F)F 48688,n1(CCCC)nc(C)c(C=CC(=O)N(CC(C)C(=O)OC)CCC)c1Cl 48689,C1(COCC)C(C)CCCN1C1(CNC(=O)OC(C)(C)C)CC1.c1cnc(C#N)s1 48690,Cc1cnoc1C(=O)NCC1(NC(C2CC(CC3CC3)C2)=O)CCC1 48691,N1(C(C2CCN(CC(C)C)CC2)=O)CCC(NC(=O)CCC(C)(C)C)C(C)(C)C1 48692,C1(C(N2CC(CC(C)C)OCC2)=O)CC(O)CCN1C(c1cc(O)cc(F)c1)=O 48693,N1(c2ncc(C(=O)OC)s2)C2CCC1C(NC(=O)NC(=O)C1CC1)C2 48694,C(CC(CNC(=O)C(C)(C)C1CCCCO1)NC(C1(OC)CC1)=O)OC 48695,N1(C(CCC=CC)=O)CCC(NC(=O)CSCC(F)F)CC(O)C1 48696,Cc1cc(C(N2CC(CC(C)NC(c3cccc(=S)n3O)=O)C2)=O)c(F)cc1F 48697,c1(OC)cccc2c(C(=O)N(CC(C)NC(=O)Cc3cncc(O)c3)C)csc12 48698,S(=O)(=O)(c1ccc2c(c1)CCCC2)N1CC2(OCCN(C(C3CC3F)=O)C2)C1 48699,c1(NC(C2CCC3(CN(C(C(C)n4cccn4)=O)C3)O2)=O)cccc2cnccc12 48700,c1(C(=O)NCC(C)NC(=O)C(O)CC2CCOCC2)cc(Cl)ccc1C(F)(F)F 48701,C1(C(N2C(C)CCC(CNC(=O)CCC3CCCC3)C2)=O)CC2CCC(C1)C2O 48702,CN1CC(NC(C2C3CC3CN2C(=O)CCc2nncn2C)=O)CC1=O 48703,C1(CNC(c2csc(Cl)n2)=O)CCN(C(=O)C=Cc2ccncc2)CCC1(F)F 48704,C(=O)(CCCC(=O)N1CC(C)(CCC(=O)Nc2cnc(F)cc2C)C1)OCC 48705,C1(OC)CCCC(CNC(C2CC(C)N2C(c2cscc2Cl)=O)=O)C1 48706,N1(C(C(C)CC2CCC2)=O)CC2CC(CNC(c3cnc(S)[nH]3)=O)C2C1 48707,c1(CN(C(CNCCCNC(C(C)OCCOC)=O)=O)C)cc(OC)ns1 48708,C(CC(C(=O)N1CCC(NC(C)=O)C1)NC(C)=O)SC.C12CCOCC1C(=O)N2 48709,c1(C(N2CCC(NC(CCSCCC)=O)(CO)CC2)=O)cc2ncccc2s1 48710,C1(N(C(COC)=O)C)CCCC(N(C)C(c2cn(C3CC3)cn2)=O)C1 48711,C1(C)(CNC(CCc2n(C)cnn2)=O)CCN(C(C23CCCCC2C3)=O)CC1 48712,CC1CC(NC(c2nncn2C)=O)CN1C(=O)CCC1CCCN1C 48713,N1(C(COC(C)(C)C)=O)CCC(N(C(=O)CC2C=CCCC2)CC2CC2)C1 48714,c1(OCC)ncc(C(N2CC(NC(=O)CCCC3CC3)CC(C)C2)=O)cc1Cl 48715,N1(C(C(C=C)O)=O)CCCN(C(c2nc(OC)c(C)s2)=O)CC1C(C)C 48716,C1(C#N)(CCC(=O)NC(C)C(C)N(C)C)CN(C(=O)OC(C)(C)C)C1 48717,C1(C(=O)NC(C(C)C)CNC(=O)CCCSC)CCOC(=O)N1 48718,CCC(C)CCC(=O)NC(C)C(C)(C)C(=O)NCCN(CC(F)F)C 48719,C1(N(C(C(C)=C2CCC2)=O)C)CCN(C(=O)Cn2ncccc2=O)CC1C 48720,C(CCC)(C(=O)NC1COCC1CNC(C1CSCCS1)=O)=CCC 48721,N1(C(c2n(CC)ccc2)=O)CCCC12CCN(C(=O)CC1CC3CCC1O3)C2 48722,C1(C)(CNC(C(C2CC2)NC(CCc2cn(C)nc2)=O)=O)CCCCO1 48723,c1(C(=O)CN2CCC3(CCC(=O)N3)C2)cc2c(cn1)OCCC2 48724,CC(CN(C)C)CC(=O)N1CCC(CC(=O)NC2CC(CN(C)C)C2)CC1 48725,Cc1cc(Br)ccc1CC(=O)NCC#CCNC(c1cc(C2CC2)nn1C)=O 48726,C1(C(N2CC(O)(C(=O)OC)C2)=O)CC2CCC1N2C(=O)COCCF 48727,CCC(CCCC(=O)NC1CCCC1)NC(=O)CN(C)C(C)C 48728,c1(CC)cc(C)c(C(=O)NCC(=O)NCCCN(C(=O)C2=CCCC2)C)o1 48729,N1(C(C2(CCCC)CC2)=O)CCC2(NC(c3cc(-c4ccc(C)s4)[nH]n3)=O)CC2C1 48730,C(=O)(C(O)CC(C)(C)C)NCCN(C(c1c(N)sc(C)c1C)=O)C 48731,C1(O)(CNC(CC2(CS(C)(=O)=O)CC2)=O)CCCN(C(c2nnc(O)nc2O)=O)C1 48732,C1(CC(C)NC(=O)CC(C)(F)F)CCN(C(C2CCCCN2C)=O)CC1 48733,c1(CC(=O)Nc2cc(Cl)c(Br)cc2O)cc2ccccc2nc1O 48734,n1(C(C)C)cccc(C(=O)NCc2cn(CCNC(C3CC(F)C3)=O)nn2)c1=O 48735,c1(C(=O)NC2CCN(C(C(C=C)O)=O)CC2)ccc(Cl)c(OC)c1 48736,CCC(C)C(O)C(C)C(=O)N1CCCC(C(=O)N(C)CC2(CO)CC2)CC1 48737,c1(C(=O)NC2CCN(C(C3C(OC)C3)=O)C2C2CC2)ccc(C)c(C)n1 48738,N1(C(c2c(OC)n[nH]c2)=O)CCC(CO)(CNC(c2c(Cl)cnn2CC)=O)CC1 48739,C1(C(=O)NCCCN(C(=O)CC(C)(C)F)C)CCCCC1(C)C 48740,C1(NC(C(C)n2cccn2)=O)C2CC3CN(C(=O)C#CC4CCCC4)C1C3C2 48741,N1(C(CCCSC)=O)CCCCCC(Nc2ncc(Br)c(O)n2)C1 48742,N1(C(c2c(OC)ccnc2)=O)CC(NC(=O)Cc2csc(C)c2)CC(F)(F)C1 48743,C(=O)(C1CC(=O)c2ccccc21)NCC(C)NC(Cc1c(C)cc(C)cc1C)=O 48744,N1(C(c2cc(C)ns2)=O)C2CCCC1CC(NC(c1c(C)[nH]c(C)c1C)=O)C2 48745,c1(C(=O)NCCOCCN(C(C(COC)(C)OC)=O)C)c(C)cccc1[N+](=O)[O-] 48746,CCCC(C(=O)OC)C(=O)NC1CN(C(c2scnc2C)=O)C1 48747,N1(C(C2CC(=C)C2)=O)CCC2(C1)CN(C(=O)C(C1CCC1)OC)CCO2 48748,c1(C(=O)NC2C(NC(Cc3cn(C)nc3)=O)CCC2)ccc2cnnc(O)c2c1 48749,C(=O)(CCC(C(C)C)NC(=O)Cn1nccn1)NCCC(=O)NCC#C 48750,N1(C(C2(CC)CCCN2C(C2CC2C2CC2)=O)=O)CC2(C1)CN(C)C2 48751,C1(CNC(c2ccnc(-n3cccc3)c2)=O)CN(C(C2CCOC2=O)=O)CCO1 48752,c1(CC(N2CCC(n3cc(C4CCCC4O)nn3)C2)=O)cc(C(=O)O)co1 48753,c1(C(N(C(C)CNC(C2CC2C(=O)OC(C)(C)C)=O)C)=O)csc(CO)n1 48754,N1(C(CCC(C)C)=O)CC2CCC(NC(c3cccc(CN=[N+]=[N-])c3)=O)C2C1 48755,CCC(C)(C)CCN=c1[nH]c(N2CC(CCOC)OC(C)C2)nc2cccnc12 48756,CC(C)C(=O)C(=O)NC(c1ccnn1C)C(N1CCC(OCCO)C1)=O 48757,N(C(=NCC1COC(=O)O1)N1CC2CC(C1)c1cccc(=O)n1C2)CCN=[N+]=[N-] 48758,C1(NC(Cc2cc(C)ns2)=O)CN(C(=O)C(O)CC(=O)OC(C)(C)C)CCC1F 48759,c1(N2CC(NC(c3cc(OC)ncn3)=O)(CO)C2)cc(C)cc(C)c1 48760,Cc1cc(C=CC(=O)NC2CC(NC(c3csnn3)=O)C23CCC3)c[nH]c1=N 48761,c1(C(=O)NC2CC(C)(NC(c3cc(C)oc3C)=O)C2)nccc2ncccc12 48762,c1(C(N2CC3C(CNC(c4cc(O)ccc4F)=O)(C3)C2)=O)ccc(I)cc1Br 48763,Cc1scc(C(N2CCC2CNC(=O)C(c2ccccc2)OCCCF)=O)c1C 48764,C1(C(N2CC(OC)C2)=O)CC(C)CN1C(=O)CCC1CC1(F)F 48765,CCC(CC(=O)NCC(C1CCN(C(c2cc(C)c(C)o2)=O)CC1)(C)C)C(C)C 48766,CC1CCCC1(C)C(=O)NC1CC(CCNC(c2csc(CO)n2)=O)C1 48767,C1(C(=O)NCC(CC)NC(C2(N(C)C)CC2)=O)CCc2cc(OC)ccc2C1 48768,C1(NC(C2CCN(C)C2=O)=O)CC2CC1N(C(c1ccccc1OC(F)F)=O)C2 48769,N1(C(c2nn(C)c(F)c2)=O)CCCC1C1CCCN1C(c1n[nH]c2c1CCC2)=O 48770,CC(C)C(C)C(CNC(=O)CCS(C)(=O)=O)NC(C1CC(OC(F)F)C1)=O 48771,N1(C(C(CC(=C)C)C)=O)Cc2ccnn2CC(NC(c2cc(CC)oc2C)=O)C1 48772,O=C1CSC2(CN(C(C34CCC(CC3)N(C(c3nocc3Cl)=O)C4)=O)C2)N1 48773,c1(CNC(C(C2(O)CCC2)NC(=O)Cc2cccs2)=O)ccc(Cl)nc1 48774,Cc1ccc(NC(=O)C(CC2CC2)NC(=O)CC2CCN(C)C2=O)cc1C#N 48775,c1(C(=O)NCCN(C(C(CC)n2cccn2)=O)C(C)C)c[nH]cc(F)c1=O 48776,c1(OC)cc(Cl)ccc1C(=O)NC1CC(NC(c2cnccc2C)=O)C12CCC2 48777,N1(CC)CC(C(=O)N2CCC(C)(NC(=O)CS(=O)(=O)CC)C2)c2ccccc21 48778,Cc1nc2c([nH]1)CC(C(N1CCN(C(C3CC4(CC4)CO3)=O)CC1)=O)CC2 48779,C=CC1CCCN(CC(=O)Nc2scc(-c3ccc(C)cc3)c2OC)C1 48780,C1(=CC(=O)NC2CC(O)CN(C(=O)CC3CCOCC3)C2)CN2CCC1CC2 48781,CC1CN(C(=O)C(C2CCCCCC2)O)CC(C)N(C(c2cc(C#N)c[nH]2)=O)C1 48782,Cc1nc(NCc2cccc3ncccc23)cc(=NCc2ccnn2C(C)C)[nH]1 48783,c1(-c2nc(C)nn2CC2(C)CCC2)cc(F)cc(Cl)c1 48784,c1(C(=O)NC2CCCN(C(C(CCC)CC)=O)CC2)cccc2c1CC(C)(C)C2 48785,C1(NC(c2[nH]cc(C)c2)=O)CC(CNC(c2cnc(C)cc2Cl)=O)C12CCC2 48786,N1(C(c2n[nH]cc2Br)C(=O)NC(CC)(C)C)CCCCC12CCN(C)C2 48787,C1(NCC)OCCC1C(=O)NCCOCCN(C)C(c1cc(C(C)(C)C)on1)=O 48788,c1(C=O)ccc(C2CC2)o1.C1(CCNC)CCCO1.C1(=O)C(c2ccoc2)N1 48789,Cc1oc2cc(C(=O)NCCN(C)C(C3(O)CC3(C)C)=O)[nH]c2c1C 48790,C1(CCOC)CN(C(=O)C(F)(F)CO)CCN1C(C1Cc2nncn2C1)=O 48791,C=CCC(C)(O)C(=O)NC(C)C(=O)NCC(C)(C)C1CCCO1 48792,C(=O)(C1CCCc2nc[nH]c21)CC=CCN=c1snc(C(=O)OC)[nH]1 48793,CC(C)CC(CCO)NC(=O)CC1CCC(NC(c2csnc2Cl)=O)C1 48794,c1(C(=O)NCCC(C)N(C(C(CC)n2cccn2)=O)C)cc(C)nc(N(C)C)n1 48795,N1(C(=O)OC(C)(C)C)CCN(c2nccn2-c2ccccc2)CC1CO 48796,N1(C(C(c2ccc(Cl)s2)C)=O)CCC(N(C)C(C2(C)CC(F)(F)C2)=O)CC1 48797,c1(CNC2CC(C(=O)NCc3cnc(Cl)nc3Cl)C2)c(F)cc(Br)cc1F 48798,N1(C(CC)=O)Cc2ccccc2C1C(=O)Nc1nc2ccccc2nc1OC 48799,C1(NC(C(CC=C)OC)=O)CC2(C1)CC(C(=O)NCC1C(C)C1C)C2 48800,C1(CC=C)CC(O)CN1C(c1occc1CNC(=O)CSCCCC)=O 48801,CC(F)(F)CC(=O)NCCN1CCC(NC(c2ccccc2Cl)=O)CC1 48802,C1(NC(C2C(CCOC)C2)=O)CCCCN(C(=O)Cn2nccc2C)C1 48803,C(CN=C(NCc1ccco1)NC(c1ccccc1Cl)C)N(CC)CC 48804,C(CCC(C)(C)C(=O)NCc1cc(Cl)ccn1)NC(C(C(=O)OCC)CC)=O 48805,C(=O)(CCCC(=O)NCC1CC(CN)C1)C(c1cccc(NC(=O)C2CC2)c1)=O 48806,N1(C(Cc2cn(C)nn2)=O)CCCC2(CCC(NC(=O)C(=O)N=S(C)(C)=O)C2)C1 48807,CC1CC2(CCN(C(=O)CS(N)(=O)=O)CC2)CN1C(C1CNC(=O)N1C)=O 48808,CC(CC(=O)N1CC(O)(C(C)(C)CNC(c2ccc(C3CCCO3)[nH]2)=O)C1)C1CC1 48809,Cc1n[nH]c(C)c1SCC(=O)NC1(CNC(=O)C(C)c2cncs2)CCCCC1 48810,CC1(NC(c2cc(C(C)(C)C)ns2)c2nnnn2CC2CC2)CC(F)(F)C1 48811,C#CCC(CC#C)C(=O)NCC1(C)CN(C(C2(C)CCC2)=O)CC1C 48812,N1(C(c2n(CCC)ncc2)=O)CC2CC1CN2C(c1c(Cl)sc(C)c1C)=O 48813,N1(C(CSCC#C)=O)CCC=CC1C(N1CC(C(C)C)C1C(C)C)=O 48814,Cc1cc(C)cc(C(=O)NC(C)CCNC(c2cnc(Cl)[nH]2)=O)c1C 48815,C1(c2ccccc2)(NC(CCc2cnn(C)n2)=O)CCN(C(=O)C=CC2CC2)C1 48816,N1(C(C2(C)COC2)=O)CCCC(CCCCNC(C23CCCC2(C(N)=O)C3)=O)C1 48817,N1(C(C(=Cc2ccccn2)C)=O)CC2CCC(CNC(C3(F)CCOC3)=O)C2C1 48818,Nc1cc(C(=O)NC2CC(CNC(c3ccc(Cl)cn3)=O)C23CCC3)cnc1N 48819,C(=O)(CS(=O)(=O)C1CCCC1)NCC1(C)CCCN1C(C1CCCC12CC2)=O 48820,C=CCCCCC(=O)NC1CC(O)CN(C(=O)CCc2ccccc2OC)C1 48821,Cc1ccc(F)c2[nH]c(C(N3CCN(C(c4cnn[nH]4)=O)CCC3C)=O)cc12 48822,C(c1ccc(C)cc1)=CC(=O)NCCO.N12CCC(CC1)C2=O.C1(C)(CC)CC1 48823,c1(C(N(CCCCN(C(C(C)NC(=O)NC)=O)C)C)=O)c[nH]c2ncccc12 48824,c1(C(N2C3CC(NC(C(C)OCC#C)=O)C2CC3)=O)c(Br)cc(F)c(F)c1F 48825,N1(C(c2cn[nH]c2)=O)CCC2(CCN(C(=O)C(O)CC3CC3)C2)C1 48826,C#CCCCCC(=O)NCc1cc(C(=O)NCC2(C3CC3)CCCO2)n(C)n1 48827,c1(C(=O)NC2C(C(C)C)CN(C(=O)C3=CCCS3)CC2)n[nH]c2ccccc12 48828,C1(NC(c2c[nH]nc2Oc2ccccc2)=O)CCCCN(C(=O)C2=C(Cl)CC2)C1 48829,C=C(Cl)CC(C(=O)NCCCN(C)OC)NC(c1ccncc1OC)=O 48830,c1(CNC(C2CCCSC2)=O)nc2c(s1)CCN(C(C1CCCN1C1CC1)=O)C2 48831,c1(CN2CC(C(=O)NCC3(C(F)(F)F)CC3)SCC2)nccc2occc12 48832,C1(NC(C2(OCC)CCC2)=O)CCN(C(=O)Cc2ccc(C)s2)CC1F 48833,CC(C)S(=O)(=O)C(C)C(=O)N1CCC(n2cc(-c3cncc(CO)c3)nn2)CC1 48834,CCC(C)C(O)C(C)C(=O)N1CC(C(=O)Nc2cnc(C)c(C)c2)(SC)C1 48835,C1(CNC(=O)NC2C(C)CCN(Cc3ccccc3)C2)CCc2scnc2C1 48836,C1(C(=O)NC(C)CCNC(c2conc2C(C)(C)C)=O)CCN(S(N)(=O)=O)CC1 48837,C1(NC(=O)Cc2csnn2)CCCCC1NC(c1cc(C(F)F)ccn1)=O 48838,C12(NC(c3c(C)nc(N(C)C)s3)=O)CCCC1CN(C(c1ccc(=O)oc1)=O)C2 48839,c1(CNC(CCOC(C)C)=O)ncccc1C(=O)NC1CCC1 48840,CCCCC(F)C(=O)N(C1CCCN(C(=O)C(C)(C)OCC)C1)C 48841,N1(C(C(CCC)(C)C)=O)CC2(C(=O)NCc3nc(C)ns3)CCC1CC2 48842,c1(NC2CCCN(C(CC(CCC)CC)=O)C2)nccc(C)c1[N+](=O)[O-] 48843,C1(C(=O)NCCOCCC#C)(CC)CCCN1C(=O)C=CCC 48844,CC1CCC(CNC(c2csc(=N)[nH]2)=O)CN1C(=O)CC1(O)CCCCCC1 48845,C(CCCCC(=O)NCC1(NC(c2csc(C)c2N)=O)CCC1)OCC 48846,CCC(CNC(c1cnn(C)n1)=O)(CC)NC(=O)Cn1ncnn1 48847,C(=O)(CC(C)CC(=O)NCC1CCN(C(c2cncc(OC(C)C)c2)=O)C1)OC 48848,c1(CC)ccc(C=CC(=O)NC2(CNC(C3(C)CC3C)=O)CCCC2)o1 48849,C1(C(=O)NCCC(C)NC(C2(CCCC)CC2)=O)CCCCN1c1ncccn1 48850,C(C)(CCC(=O)N1CC2C(NC(C3CC(=O)N(C4CCCCC4)C3)=O)C2C1)OC 48851,CCC(CC(=O)NC(CN(C)C(c1cccc(C(C)C)n1)=O)CC)OC 48852,C(=O)(C1CCCn2nccc21)NCC(COC)NC(c1ccc(F)cc1F)=O 48853,N(C1CCc2cccc3cccc1c23)C1CCN(N(C)C)CC1.C(=O)NCC 48854,c1(OC)c(C)cc(C(=O)NCCC(C)NC(C2(C(C)(C)C)CCC2)=O)cc1Cl 48855,C1(O)(CCNC(c2n(CC)c(O)nc2)=O)CCN(c2ncncc2C#N)CC1 48856,c1(C(N2CCC(NC(C(C)(C)F)=O)C2C(C)(C)C)=O)ncc(N)cc1Cl 48857,CCCC(C#N)C(=O)N1CCN(C(c2ccncc2Cl)=O)C(C2CCC2)C1 48858,c1(C(=O)NCC2N(C(CN(C)C(c3ccccn3)=O)=O)CC2)cnn(C2CC2)c1 48859,N1(C(c2ccc(CC)[nH]2)=O)CCOCC1CNC(=O)C(c1ccc(OC)cc1)O 48860,N1(C(CC(=O)NCC#C)=O)CCC2(CCC(CNC(=O)Cc3cnc[nH]3)O2)CC1 48861,C1(NC(C(C)CO)=O)CN(C(=O)C(C)(C)c2ccn(C)n2)CC2CCCC12 48862,c1(C(=O)NCCC(CNC(CCn2c(C)ncc2)=O)O)cncc2nc(O)[nH]c12 48863,c12cc(nn1C)C(=O)NC2.C1(C(N2CCC2C2CCCC2)=O)(OCC)CCCC1 48864,C1(CNC(C2(COC)CC2)=O)CCN(C(c2ccc(C(C)(F)F)cc2)=O)CC1C 48865,CCCC(C)(O)C(=O)NCC1CCCN(C(c2cc(C(F)(F)F)nn2C)=O)C1 48866,N1(C(C(Cc2ccoc2)NC(C2OCC(C)(C)C2)=O)=O)CCC(C2(C)CC2)CC1 48867,C1(CC(=O)N(C(C)C2CC2)CC)CN(C(=O)CCCC2CCCO2)CCO1 48868,c1(CC)ccc(OCC(=O)NC2(CO)CN(C(=O)CCn3cnnn3)C2)cc1 48869,c1(-n2ccc(C(=O)NCC(C)N(C(=O)CC(C)SC)CC)n2)ccc(F)cc1F 48870,C1(O)(CCNC(C2COCCC2(F)F)=O)CCCN(C(=O)CCc2cnoc2)C1 48871,C1(NC(Cc2ccc(C)nc2)=O)CCN(C(=O)CC2OCCCO2)CC1(C)C 48872,c1(CNC)cccc(NC(=O)C(N2CC(CN)C(C)C2)=O)c1 48873,N1(C(c2c[nH]cc(C)c2=O)=O)CC(NC(=O)Cc2nc[nH]n2)C2(CCCC2)C1 48874,C(=O)(C(F)(F)C(F)(F)F)N(C1CN(C(=O)CC2CCC(C3CC3)O2)C1)C 48875,CC(C)C(C(=O)NOCCCN(C)C)C(C)NC(=O)CP(C)(C)=O 48876,C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NCC1(NC(CC(CC)C(F)F)=O)CCOC1 48877,C=CC(C)(CCOC)C(=O)NC1CCC1C(=O)NCc1ncoc1C1CC1 48878,C1(C(=O)N(C2CCCCCC2)CCNC(C2(O)CCC2)=O)CC2CCCCCC12 48879,N1(C(C(C)NC(C)=O)=O)CC(NC(=O)C(C)Cc2c(C)n[nH]c2C)C(C)(C)C1 48880,c1(CCC)cc(C(N2CC(C(C)(C)O)(CNC(C3(F)CC3C)=O)C2)=O)no1 48881,c1(C(N(CCOCCNC(C(CCC)C#N)=O)C)=O)c(F)ccc(F)c1Cl 48882,C#CCCC(O)C(=O)N1CCCN(C(C2CCC(F)(F)C2)=O)CC1 48883,Cc1cc(C(N2CCC(C(=O)O)(C(C)C)C2)=O)nc(O)c1 48884,C1(CNC(=O)CCN2CCCCC2)COCCN1C(=O)COC(F)(F)F 48885,C#CCCCCCCC(=O)NCC1(NC(=O)Cc2nccc(OC)n2)CCOC1 48886,C1(CC=C)(C(=O)NC(C(=O)NCCSCCOC)C2CC2)CCOC1 48887,CC(C)CCC(=O)N1C(CNC(c2ccc(N3CCCC3=O)cc2)=O)CC2CC12 48888,N1(C(C2CCSCC2)C(=O)Nc2ccc(F)cc2)CCC(c2nncs2)CC1 48889,C1(CNC(CC)C(N)=O)(CO)CC(NC(=O)OC(C)(C)C)C1(C)C 48890,c1(C(=O)NC2CCC(C)(CNC(CC3(CSC)CC3)=O)C2)cc(C#N)[nH]c1C 48891,C#Cc1ccc(C(=O)NC2CC(C)(NC(c3cccc(C(C)C)n3)=O)C2)cc1F 48892,N(C(=NCCCN1CCOC1=O)NCCOc1ccc(Cl)cn1)CC(C)C 48893,C=C=CCCC(=O)NC(C1CCN(C(c2nccc(C(F)(F)F)n2)=O)C1)(C)C 48894,c1(C(=O)NC(C2CCCN(C(c3csc(C4CC4)n3)=O)C2)C)c(O)cccc1Cl 48895,N1(C(C(CC(=C)C)OC)=O)CCC(NC(C2CCN(C)C2)=O)C(C)(C)C1 48896,CCCCCC(O)CC(=O)N1CC2CCN(C(c3cc(Cl)ccc3Cl)=O)C(C2)C1 48897,C1(CNC(C(COC)N(C)C)=O)CCC2(CCC2)CN1C(=O)C(O)C(C)(C)C 48898,Cc1cccc2c1C(NC(C1(C(=O)O)CCSC1)=O)CC2 48899,c1(C(C)(C)C#N)ccc(C(N2CC(NC(C3(Cl)CC34CCC4)=O)C(O)C2)=O)cc1 48900,n1(C(C)C)ncc2cc(C(N3CC4CC3CN(C(C3CC(O)C3)=O)C4)=O)cnc12 48901,C1(C(C)NC(C2(CO)CCC2)=O)CCCCN1C(=O)CSc1cccc[n+]1[O-] 48902,c1(OC)cc(C(=O)NCC(CC(C)C)NC(=O)C=CC2CCOC2)n(C)n1 48903,N1(C(CC(C)NC(C)=O)=O)CCCC(NC(C2CCC(CC(C)C)CC2)=O)CC1 48904,N1(C(C2C(C#N)C2)=O)CCc2c(CNC(=O)CC3=CCOCC3)cccc2C1 48905,c1(C(=O)OC)cn2c(n1)CCCN2C(=O)Cc1nc(Cl)n(C)c1C 48906,CC(C)CCCCC(=O)N1CCCC1C1(O)CN(C(=O)C(=O)NC(C)C)C1 48907,C1(COC)(NC(=O)CCn2cncn2)CCN(C(=O)COc2cn[nH]c2)C1 48908,C#CCC(C)(CC)C(=O)NC1CC=CCC1C(=O)NCC1(C)CC(C)C1 48909,Cc1cc(NC(=O)C(=O)NC(C2COCCO2)C)ccc1NS(=O)(=O)C1CC1 48910,C(=O)(CCC1=CCCCC1)N1CCCC(N(C(C2CC(SC)C2)=O)CCO)C1 48911,c1(OC(C)C(=O)NCCC(C)N(C(=O)CNc2cccnc2)C)ccccc1Cl 48912,C(=O)(C1CCc2nccn21)NCC1CC(OC)CN1C(c1cc2occc2[nH]1)=O 48913,N1(C(=O)CCc2ccon2)CCC(NC(C2CC(n3ccnn3)C2)=O)CC(O)C1 48914,C(CCCC(=O)NOCCO)N(C)C(c1ccc(F)c(O)c1)=O 48915,C(C)(C)(CCCC(=O)N(CC(C)C(C)C)C)NC(c1c(C)ccnc1)=O 48916,C1(NC(c2c(OC)cnc(Cl)c2)=O)CC2CCC(C1)N2C(C1(C#N)CCC1)=O 48917,N1(C(c2cnc(SC)s2)=O)CC2(CCN(C(c3ccncc3N)=O)CC2)CC1C 48918,O=S(=O)(c1cnccc1N1CC2C3CCC(C3)C2C1)NC(CF)CF 48919,C1(NC(CC2(C)CCOCC2)=O)CC(C(=O)NCc2nnc(O)o2)=CC1O 48920,c1(C(=O)OC)ccc(=NCC2CCCN(C(=O)C(C)P(C)(C)=O)CC2)[nH]c1 48921,Cc1ccc2occ(C(=O)NCC3CN(C(C4CC(O)C4)=O)CC(C)(C)O3)c2c1 48922,N1(C(c2cc(C)c(F)c(C)c2)=O)CCN(C(=O)C(O)C(F)F)C2CCCC12 48923,c1(N2CCN(C(C(=O)NCC3C(C)(C)C3(F)F)=O)CC2)ccc(C#N)cc1Cl 48924,C1(CNC(N(CCCC)Cc2ccco2)=O)CCC(Oc2ccncc2)C1 48925,C(C)(CC(=O)N(C1CCN(C(=O)Cc2csc(NC=O)n2)C1)CCO)OC 48926,Cc1snnc1C(=O)NC(CC1CCOCC1)C(=O)NCCC(C)N(C)C 48927,Cc1nc(C(=O)NC2CC(C(F)F)(NC(c3nsnc3O)=O)C2)cn(C)c1=O 48928,CC1CCCn2ncc(C(=O)NCC3(O)CC(NC(c4ncc[nH]c4=O)=O)C3)c21 48929,N1(C(CCCOCC=C)=O)CCC(C)(CCNC(=O)COc2ccon2)C1 48930,C#Cc1ccc(OC)c(C(=O)NC2CCN(C(=O)C(C)C(F)(F)F)C2)c1 48931,CCCCCCCCCC(CC)C(=O)N1CC(C2CN(C(=O)CCCOC)C2)C1 48932,c1(CC(C)C(=O)OC2CCN(c3ccc(F)cc3)C2=O)ccc(Cl)cc1Cl 48933,CCCC(CCCNC(=O)C1=CCSC1)NC(=O)CC(CC)C1CCC1OC 48934,C1(C(=O)NC(C=C)C)CCC(C)N(C(c2cnc(CC)cn2)=O)C1 48935,c1(CC)cccc(NC(C2(C)CCCN2C(=O)C(c2ccc(C)o2)C)=O)c1F 48936,N1(Cc2cn(CCC=C)nn2)CCCCC(C(=O)N(C)C)C1 48937,C12(NC(c3cnco3)=O)CCN(C(c3ncoc3-c3ccco3)=O)CC1C2 48938,C1(C)(C(=O)NC(C)Cc2ccco2)CC12CCN(c1cc(C#N)ccn1)CC2 48939,N1(C(c2scc(COC)c2)=O)CC2CCN(C(=O)CCCCCF)CC2C1 48940,N1(C(C2C(C(N)=O)CC2)=O)CCCC(CNC(C2(F)CC2c2ccccc2)=O)C1 48941,Cc1ncccc1CCC(=O)N(CC(O)CN(C)C(C1C=CCS1)=O)C 48942,N1(C(CNC(c2n(C)c(S)nn2)=O)=O)CCC2(CC1)CC2(C)C(=O)NCC1CC1 48943,C12(C(=O)NC(C(C)(C)NC(Cc3c(C)n(C)nc3)=O)C)CC(CO)(C1)OC2C 48944,C(=O)(CCCCCC(C)O)NCCC1(NC(c2c(CCC)cccc2)=O)CC1 48945,C(=O)(C(C)(C)CCC#N)NCC(C)(C(C)C)NC(CCc1ccc(C)s1)=O 48946,c1(CC)cccc(NC(=O)C(Cn2cncn2)NC(c2nonc2N)=O)c1C 48947,C(c1csc(C(F)(F)F)c1)=CC(=O)NCC(CNC(C1(F)CC1)=O)OC 48948,O=C(C(=O)C(F)(F)F)NCc1cn(C2CCN(C(=O)C(O)c3ccsc3)C2)nn1 48949,N1(C(C=NOC)=O)CC2(CC(NC(c3cc(Cl)ns3)=O)c3nccn32)C1 48950,CC(C)(C)C(=O)NCCCC(=O)NCC1(NC(=O)Cn2ccc(=N)[nH]2)CC1 48951,C1(CC(=O)NC2CCC(CNC(C(CC)N3CCCC3=O)=O)C2)CCCOCC1 48952,N1(C(C2(C3(C)CC3)CC2)=O)CC(C(=O)NC2(C)CCSC2)C2(CCC2)C1 48953,N1(C(C(COC)(C)C)=O)CC2(C)CC1(C(=O)NC(C)CCC1CCCO1)C2 48954,C(=O)(C1(C)CCOc2ccccc21)N(CCNC(C(CCCC)CC)=O)C 48955,C1(C(N2CC(CCNC(=O)CSc3ccccc3Cl)C2)=O)CCCC2CCCN12 48956,C(=O)(C(CCCC)NC(C1CCCS1)=O)N1C(C=C)CCC1 48957,Cc1nc(C(N2CCCC(NC(=O)C(C)Cc3ccnn3C)C2)=O)c(C)s1 48958,C#Cc1cccc(C(N2CCC(CN(C)C)C2)C(=O)NC2CCOCC2)c1 48959,C#CCCCCCCC(=O)N1CC2(CC(CC(N3CCOCC3C3CC3)=O)C2)C1 48960,N1(C(C2C3COCC23)=O)CCC(CNC(CC2CCN(CCC)C2)=O)CC1 48961,C12(C(=O)NCC3CC(NC(C4C(C(N)=O)CC4)=O)C3)CCC(OC(F)F)(CC1)C2 48962,NC(=O)N=Nc1ccc(C(=O)NCC2CC(NC(C3CCCN3C=O)=O)C2)cc1 48963,n1(CC)ncc(C(c2nnnn2C2CCC2)Nc2ncccc2CCOC)c1C 48964,Cn1nc(-c2nc(C3CC34CC4)nn2C2CCCSC2)c2c1CCCC2 48965,N1(C(CC(CNC(=O)CC=C(Cl)Cl)OC)=O)CC(C)(C2CCC2)C1 48966,N1(C(Cc2ccc(C)o2)=O)CC(NC(c2cncn(C)c2=O)=O)CC1(C)C 48967,c1(OC)ccc(F)cc1CC(=O)N(C)CCNC(=O)Cc1cccc(Br)c1 48968,CC1CN(C(C2(C)CCCN2C)=O)CCC1C(N1CCCC(O)(C(N)=O)C1)=O 48969,n1(CC=C)cccc1C(=O)NCC(C)NC(=O)Cc1ccoc1C 48970,Cc1noc2nc(-c3ccco3)cc(C(=O)NOCC(=O)N(C)O)c12 48971,C1(NC(C2CN(C)C(=O)C2)=O)CC2CCCC(C1)N2C(c1cccn1C)=O 48972,C1(C(N(C(CNC(C(C)=CC)=O)C)C)=O)CCCCCS1(=O)=O 48973,c1(OC)cc(F)c(C(=O)NC2CC(CNC(c3ccnc(Cl)c3)=O)C2)cc1F 48974,c1(C(N(C(C)CNC(=O)C(F)Cc2ccccc2)C)=O)cccn2ccnc12 48975,C(c1ccccc1)=C(C(=O)NC(C)CN(C)C(c1cccnc1)=O)C#N 48976,n1(CC)ncc(CNC(C2(C)CCN(C(=O)CN=[N+]=[N-])C2)=O)c1C 48977,CC(C)(CCCF)NC(C1CC2CC2N1C(=O)CCCC1CC1)=O 48978,C1(C(=O)NCCOC(C)=O)CCN(C(c2cc(C)c(C)cn2)=O)CCO1 48979,c1(C(N2CCC(O)(CNC(CN3C(C)CCC3)=O)C2)=O)cc2scnc2[nH]1 48980,Cc1ccc(C(C)OC(c2scnc2C2CC2)=O)s1 48981,N(C(=NCCOCC1CC(SC)C1)NCC(C)C)C1CCN(C(=O)OCC)CC1 48982,C1(C(C)(C)C)(CNC(CC=C)=O)CCN(C(=O)Cc2ccnc(OC)c2)C1 48983,N1(C(COc2ccc(CC)cc2)=O)CCCN(CCNC(=O)C(F)CC)CC1 48984,C(=O)(CCCCC(C(F)(F)F)NC(=O)NCC1COC2(CCCC2)O1)OC 48985,N1(C(CC(C(=C)C)O)=O)CCCN(C(c2cnc(C)s2)=O)CC1CO 48986,C#Cc1ccccc1CC(N1CC(CNC(=O)CC(=C)Br)CC1C)=O 48987,c1(CN(CCCNC(c2ncccc2C2CC2)=O)CC)ccc2n[nH]cc2c1 48988,NC(CCC1CC1)C(=O)N1CC(N2CCCC2)C1 48989,Cn1cc(NC(=O)C(=O)NCC2(NC3CCCC(C(F)(F)F)C3)CCC2)c(O)n1 48990,C1(NC(C2N(C)C(=O)NC2)=O)CC2CN(C(C3CCOC(=O)CC3)=O)CC2C1 48991,C(C(C)(C)CC(=O)N(CCCNC(C1CCCN1S(C)(=O)=O)=O)CCO)OC 48992,c1(C(N2C(CNC(CC=CCC)=O)CCCCC2)=O)ncc(Cl)c(N)c1Cl 48993,c1(NC(C23C(CN(C(c4cc(OC)c(F)cc4)=O)C2)C3)=O)ccc(F)cc1C#N 48994,n1(CC)c(C(=O)NCCN(C2CCCCC2)C(=O)CCOC2COC2)cnc1O 48995,C12CCCC(C1)CNC2.c1(C(=O)NC2CN(C(C)=O)C2)cnnn1C1CC1 48996,C(=O)(C(C(C)C)C(C)C)NC1(CCNC(c2c(C)cc[nH]2)=O)CCC1 48997,N1(CCN(C(CC2ON=C(C)C2)=O)C)CCN(C(=O)C=CBr)CC1 48998,C(C#CCN=c1[nH]ccc(=NC2CCN(C3CCCCC3)C2)[nH]1)OC 48999,Cc1cc(Br)cc2c1CN(C(=O)Nc1cnc3c(c1)CCOC3)CC2 49000,CC1ON=C(C(=O)NCC2CN(C(=O)C(N)=O)CCO2)C1C 49001,CCC(C)C(C(=O)NC(C)CN1CCN(C(=O)CC2CC(C)C2)CC1)NC(N)=O 49002,N1(C(C(C)C2CCC2)=O)CC2CCC(C1)C2CNC(=O)C(O)CC(F)(F)F 49003,C1(C(=O)NCC2=NOC(C)C2)CCCCCC1NC(C1C=CCS1)=O 49004,C12(NC(c3cnco3)=O)CCCC1N(C(c1cc(-c3ccccc3)co1)=O)CC2 49005,C12(NC(c3nn(C)c(F)c3)=O)CCOCC1CN(C(c1csnn1)=O)C2 49006,C=CCC(C(=O)NC(C1(O)CN(C(c2cccc3ncsc23)=O)C1)C)C(C)C 49007,N1(CC(=O)NC2(CNC(c3c(C)[nH]cc3)=O)CCC2)CCC(=O)NC1=O 49008,c1(C(N2CC(NC(c3c(CC)onc3)=O)C3(C2)CC3)=O)ccc2n[nH]cc2c1F 49009,C1(CCC)CCCC1C(=O)NCCCOCCCNC(=O)CCCNS(C)(=O)=O 49010,C1(C(=O)NC2C(NC(COCCCC)=O)COC2)Cc2ccccc2S1 49011,CC1CN(C(=O)CSCC(N)=O)CCC1N=c1[nH]c(Cl)ncc1CO 49012,CS(=O)(=O)c1cc(C(=O)NC2C=CCN(C(=O)Cc3nc[nH]n3)C2)cs1 49013,c1(C(=O)NC2(c3ccccc3)CCN(C(C=CSC)=O)C2)cc(C)nnc1O 49014,C1(C(=O)NCC(CC)NC(=O)CCc2cn(C)nn2)CCCC1c1ccccc1 49015,C1(N(C2CCOCC2)C(=O)Cc2ncccc2F)CCCCN(C(=O)CCCF)C1 49016,C(=O)(C(C)(C)C#N)NCCC1(C(=O)NC(C(C)C)CO)CC1 49017,c1(C(N(C2CCCC(NC(=O)C(C)(C)C)C2)C)=O)cc(C2CC2)cc(Cl)c1 49018,N1(Cc2c(C)nccc2)CC2(CCC(C(=O)Nc3oncc3C#N)O2)C1 49019,Cc1nn(CC(N2CC3CC2CC3CNC(c2csnc2Cl)=O)=O)cc1[N+](=O)[O-] 49020,C(CCCCC(=O)N(C(C)CNC(C1CC(OC)C1)=O)C)=CC 49021,C(C(C)(C(C)C)NC(=O)COCCOC)NC(c1c(OC(CC)C)cccn1)=O 49022,CC(N=[N+]=[N-])C(=O)N1CC(CC(F)C(=O)NCC(c2ccccc2)F)C1 49023,CC1CCCC=C1C(=O)NC1CCN(C(=O)CC(F)(F)C(F)F)CC1(C)C 49024,c1(OC)cc(C(=O)NCC(O)CNC(C23CC(CO)(C2)OC3C)=O)cc(OC)n1 49025,c1(CNC(C(N2CCC(CCC(=O)OCC)C2)=O)=O)ccc(F)cc1CC 49026,N1(C(C2N(C(c3c(C)c[nH]c3)=O)CC2)=O)CCC2(CCCO2)C1 49027,C=CC1CCN(C(C2CCN2C(=O)C(C)SCC)=O)CC1 49028,C(CCC(C)C)(C(=O)N(C)CCc1ncccn1)NC(C1C(CCC)CCC1)=O 49029,CCS(=O)(=O)C=CC(=O)N1CCC(C)(C)C(CNC(c2cccn2C2CC2)=O)C1 49030,C1(OCC)CC(CNC(=O)CNC(=O)Cc2cc[nH]n2)C1 49031,C(c1cn(C)cn1)=CC(=O)NC(C(=O)NC(c1onc(C)n1)CO)CO 49032,C(=O)(CC1=NN(C)C(=O)C1)NCC1ON=C(C(=O)N(C2C(C)C2)C)C1 49033,N1(C(c2c(CC)cns2)=O)CC(O)CCC1C(=O)NCCn1ncnn1 49034,C(=O)(NNC(=O)C1CCCS1)NC(Cc1cc(C)[nH]n1)C 49035,C1(N=[N+]=[N-])(C(N(C)Cc2onc(CC)n2)=O)CCN(C(C2C=CCS2)=O)C1 49036,N1(C(C(CC)(C)O)=O)CCCCC2(C1)CN(C(c1nn(C)cc1C)=O)C2 49037,c1(C(=O)NC(CCNC(C(CCCC)O)=O)(C)C)cc(=O)c2cc(F)ccc2o1 49038,C1(C2CCCN(c3ccccn3)C2)(C(C(=O)O)C(=O)N2CCC(CO)CC2)CC1 49039,Cc1cc(=NCC2CC(C)CC(C)C2)[nH]c(=NCCS(=O)(=O)C(F)(F)F)[nH]1 49040,N1(C(CC2(CSC)CC2)=O)CCOCC(CC(N2CCC(C)(C)C2)=O)C1 49041,C1(C(=O)NC(C2CCN(C(=O)Cc3ccccc3)C2)C)C2CC3C(C2=O)C13 49042,CCCCCC(O)C(=O)N1C(C)C2CC1C2NC(C1(C(F)(F)F)CCCCC1)=O 49043,c1(C(N(C2CCCN(C(=O)C=C3CC3)CC2)C)=O)ccc(N)c(Br)n1 49044,CCC(C)(C)CC(=O)N1CCOC(C)(CNC(=O)CC(C)OC)C1 49045,c1(C(=O)NCC2(NC(c3ccc4c(c3)NCC4)=O)CCC2)cnc2[nH]ccc2n1 49046,N1(C(C(C2CCOCC2)C)=O)CCOCC(CNC(C2CC(=O)N(C)C2)=O)C1 49047,c1(OC)ncc(Br)cc1CN(C1CCN(C(C2CCN(C)C2)=O)C1)C 49048,C=CCC(CC(C)C)C(=O)N1CC(NC(C2(C#N)CC(C)C2)=O)CC(C)(C)C1 49049,C1(C2CCOCC2)(C(=O)NCC2N(C(CCCN(C(C)C)C)=O)CC(O)C2)CC1 49050,N1(C(CCCC)=O)CC(=O)NCC1C(N1CCCC(C)(CCC)C1)=O 49051,Cc1sc(O)nc1C(=O)NCC1CCCN(C(C2(N3CCCC3)CC2)=O)C1 49052,CC(C)CC(C)CC(=O)NC1(C)CCN(C(C2(C#N)CC2)=O)C1 49053,c1(C(=O)NCC(CNC(C(CN(C)C)N(C)C)=O)(C)C)cnc2ncccc2c1 49054,C1(C(=O)NCc2cnc(C)s2)CNC(=O)CN1C(c1n[nH]c2c1CCC2)=O 49055,c1(C(=O)NCCCN(C(C)C)C(C2CCCCC2(F)F)=O)cccc2occc12 49056,C(C(C)(O)CC(=O)NC(CNC(c1cc(C(N)=O)ccc1C)=O)CC(C)C)OC 49057,N1(C(Cc2ncc(C)s2)=O)CCOC(CNC(C2CN(C3CCCCC3)C2)=O)C1 49058,CC#CCCCC(=O)NC1CCC1CNC(c1ncn(CC)n1)=O 49059,CCC(CC(=O)NC1CCCC1NC(c1c(C)cnnc1O)=O)C(C)(C)C 49060,C(=O)(CC(C)C)NC(C(=O)N(CCOC)CCOC)c1cccs1 49061,C1(C(=O)NC(C2CCCC2O)C)C=CCN(C(=O)CC2CC(=O)NC2=O)C1 49062,N1(C(=O)OC)CCCC1C(=O)N(C1CC(NC(c2cn(C(C)C)cn2)=O)C1)C 49063,c1(CN2CC(CNC(C3(CC)CCNC3=O)=O)OCC2)c(F)cccc1Cl 49064,Cc1ccc(C)c(C(=O)NC2CC3CC2N(C(C2(O)CC2(C)C)=O)C3)n1 49065,C(=O)(C#CC1(C)COC1)N1C(C)CCC(C(=O)NC(CC)CO)C1 49066,C1(CNC(=O)CCCC2CCC2)CC2(CCC2)CN1C(=O)Cc1ccncc1Cl 49067,N1(C(CNC(CCC)=O)=O)CC(F)CC1CNC(c1c(C)ncn1C)=O 49068,c1(C(N2CCC(C)(CCNC(CCOC(C)=O)=O)C2)=O)cnc2ccncc2c1 49069,n1(CCC(=O)NC2CC(NC(CN3CCC(C)(C)C3)=O)C2)cc(S(N)(=O)=O)cn1 49070,C(=O)(NNc1cc(F)c(F)cc1Br)NCc1c(CC)onc1C 49071,c1(CNC(c2csc(CO)n2)=O)cccc(NC(C2CCC(O)C2)=O)c1 49072,N1(C(C2N(C(CNC(=O)NC)=O)C(C(C)C)CC2)=O)CCOCC1C(N)=O 49073,CS(=O)(=O)c1cscc1C(=O)NCC(CO)NC(C1(F)CC=CCC1)=O 49074,c1(C(=O)NC2CC(CCC(=O)N3CC(C(F)(F)F)C3)C2)cnn2ccccc12 49075,c1(C(=O)O)cc(S(=O)(=O)N2CCC(O)(C3CC3)C2)cc2c1OCO2 49076,CC(C)CC(C)(O)C(=O)N1CCCC(CNC(=O)C#CC2CCC2)C1 49077,Cn1ncc(CC(=O)NC2CCC(NC(c3ccon3)=O)C2)n1 49078,c1(OC)ccc2c(c1)C(NC(=O)NCC1(SC)CC(C)(C)C1)CCC2 49079,CCC(C#N)C(=O)NC1CC(CNC(=O)C(c2ncccc2F)(F)F)C1 49080,C(=O)(C(CNC=O)c1ccccc1)NC(CNC(C(C)C1CC1)=O)CO 49081,CC1(C(N2CCCC(O)C2)=O)CCCN(Cc2nc(Cl)sc2Cl)C1 49082,c1(C(=O)NC(CN(C(c2c(CC)non2)=O)CC)CC)coc2ccccc12 49083,c1(C(C(=O)NCCOCC)N(c2ncc(Cl)s2)C)ccc(C#N)cc1 49084,c1(C(N2CC3(C(NC(C(CCC)C)=O)CC3)C2)=O)ccc2cc(C)cn2c1 49085,n1(CCC(=O)NC2CCN(C(c3c(C)ncnc3)=O)C2)cc([N+](=O)[O-])nc1C 49086,c1(C(N2C(CCC(=O)NC3CCN(CC)C3=O)CCC2)=O)ncc2ccccn12 49087,C1(C2CN(C(C34CCCCC3C4)=O)C2)(NC(c2cc(OC(C)C)ncc2)=O)CC1 49088,N1(C(c2c(C#N)ccs2)=O)CC(CNC(=O)CCSC(F)(F)F)C(F)(F)C1 49089,C(C(=O)NCC1(NC(c2cnn(C(C)(C)C)c2C)=O)CC1)(C(C)C)SC 49090,c1(CNC2C(CC)C2)ccc(S(=O)(=O)NCC2(c3ccon3)CCC2)cc1C#N 49091,C#CCC(C)(C(=O)NCc1nccnc1CC)NC(=O)C(=O)NC 49092,C1(c2nnc(N(CCC)CCC)n2CC2CC2)CCc2c(cnn2C)C1 49093,C(=O)(C(F)(F)C(F)(F)F)N1CC(NC(c2c(C)ncs2)=O)C(C)C1 49094,C(=O)(C(C)(C)C(C)O)NC1(COC)CCN(C(c2ccc(NC)cn2)=O)C1 49095,c1(OC)ccc2cc(C=CC(=O)NC3CCN(C(=O)C(C)C)C(C)C3)ccc2c1 49096,C#Cc1ccc(CNC(C2(NC(=O)CC3CCSC3)CC2)=O)cc1 49097,C#Cc1ccc(C(=O)NC(C(N2CC3CC3(COC)C2)=O)C2CCOC2)c(C)c1 49098,CCCCCS(=O)(=O)CC(=O)N1CCCC2(NC(c3ccc[nH]3)=O)CC2C1 49099,O=C(CCC(CF)CF)NC1COCC1CNC(c1cncc([N+](=O)[O-])c1)=O 49100,CCCCC(C(=O)NC1CCC(CCC(=O)N(CCC(=O)OC)CC)C1)C(C)C 49101,C(=O)(CS(=O)(=O)C(C)C)N(C)CC1CCN(C(c2c(CCC)nco2)=O)CC1 49102,C(N(C)N1CC2(C=Cc3ccccc3O2)C1)C1(SCC)CC1 49103,c1(NC2CC(C)N(C(c3cccc(C4CC4(F)F)c3)=O)C2)ncc2ncnc-2[nH]1 49104,c1(C(=O)NCCCCC(CO)NC(C2CC(OC)C2)=O)cccc2c1OCC2C 49105,C1(NC(=O)C(F)OC(F)(F)F)(CO)CCCN(C(C2(Cl)CC2)=O)C1 49106,c1(C(=O)NC(C(=O)NC2(C(C)C)CC2)Cn2cncn2)c[nH]nc1[N+](=O)[O-] 49107,c1(OC)nc(N2CC3(CCN(C(c4cncc(C)n4)=O)C3)C2)ncc1C#N 49108,NCC(CNCC(=O)NCCOCc1ccccc1)C(F)(F)F 49109,CC1C(NC(c2cnn(C3CC3)c2)=O)CCCN1C(=O)Cc1cc(F)ccc1F 49110,Cc1nc(C(=O)NCC(CO)NC(C2CCC(=O)N2)=O)co1 49111,N1(C(c2c(C(=O)OC)cco2)=O)CCC2(NC(=O)CC3CCCO3)CCCC12 49112,c1(OC)ccc(C(N2CCC(NC(c3ccnc(O)c3)=O)C(O)C2)=O)cc1O 49113,C(=O)(CC(O)C(C)C)N1C(C)(CNC(C2(OC)CCSC2)=O)CCC1 49114,C1(C(=O)NC2(CNC(=O)C(C)C)CC(OC)C2)CC(C)(C)CO1.c12cccc(c1)N2 49115,c1(C(=O)NC(CC)CNC(=O)CC2COC(=O)C2)nnc2n1CCCCC2 49116,C(c1ccc(S(C)(=O)=O)o1)=CC(N1C2C(NC(C#CC3(C)CC3)=O)CC(C2)C1)=O 49117,C(C(=O)NNC(=O)c1ccc(I)c(Br)c1)c1cccc(C)c1 49118,CC1CCCCC1(CNC(c1ccc(=N)[nH]c1)=O)NC(=O)CSCC#N 49119,N1(C(C=CSC)=O)CC(CO)C(C(F)(F)F)C1.c12cc(on1)CNC(=O)C2 49120,c1(OC)ccccc1C(=O)NCC1(F)CC(NC(c2conc2C2CCC2)=O)C1 49121,C1(NC(CCOC(CC(C)C)C)=O)CN(C(=O)CNS(C)(=O)=O)CC1C(F)F 49122,N1(C(c2c(C)ncn2C)=O)C2CCC1CN(C(=O)Cc1ccncc1Cl)C2 49123,CC1CC(CNC(C2(C)CCSCC2)=O)CN(C(=O)CCc2cn(C)nn2)C1 49124,C1(CNC(C=CC=CCC)=O)CCCC2CN(C(c3ccc(CC)cc3)=O)CC12 49125,N1(C(C(COC)OC)=O)CC2CC(NC(c3sc(C(C)C)nc3C)=O)CC1C2 49126,N1(C(C(CC)C)=O)CCN(C(C23COCC(C2)C3)=O)CC1CC1CC1 49127,c1(CC)cc2c(CC(=O)NCC(CC)NC(C3(C#N)CCOCC3)=O)csc2s1 49128,c1(NCC2CCCN(CCC(=O)OC)C2)cc(OC)ccc1[N+](=O)[O-] 49129,C1(NC(c2c(OC)cccc2)=O)CCCN(C(=O)C(=O)CC(C)C)C1C 49130,C1(CNC(c2cccc(O)c2F)=O)CC2CN(C(C3CC4CCC3O4)=O)CC12 49131,c1(C(N2C(COC)(CNC(c3occc3C)=O)CCC2)=O)csc(=NC2CC2)[nH]1 49132,C(=O)(C1CCSc2ccccc21)NC(CC=C)CNC(=O)CCCC(=O)OCC 49133,C(=O)(CCC(C)(C)C)N1CCC(C)(CC(N2CC(C)C(CO)C2)=O)C1 49134,C(=O)(C#CC1CCOC1)NCC(CC)NC(c1ncsc1S(N)(=O)=O)=O 49135,c1(C(=O)OC)ncc[nH]c1=NCC1(NC(c2cnc(C(C)O)s2)=O)COC1 49136,C1(CC)(CNC(C2(CC(=O)C=CC(=O)NC3CCSC3)CC2)=O)CCCCC1 49137,N1(C(C2C(NC(=O)CC3CC4(CC4)C3)C=CCC2)=O)CCc2ccsc2C1 49138,c1(C(N(CCOC)CCNC(C2CC(C)(C)C2)=O)=O)cc(F)ncc1OC 49139,c1(C(=O)NCC2CCC(C(N3CC(C)(O)C3)=O)O2)occ2c1CCC2 49140,c1(NC(C(c2ccco2)NC(COC(CC)CC)=O)=O)ccc(F)cc1O 49141,N1(C(C(C)c2ccsc2)=O)CCCC(CN(C)C(c2cnc(N(C)C)nc2)=O)C1 49142,C1(C)(c2cn(C(C(=O)OC)C)nn2)CCCN1C(=O)CO 49143,Cc1[nH]c(C#N)cc1C(=O)NC1(C)CC(NC(C23CCCC2C3)=O)C1 49144,c1(OC)cnc(C(=O)NC2CCCC2NC(=O)CC#N)cn1 49145,CC(C)(C)C(O)C(=O)N1CCCCCC1CNC(c1cnc2sccn12)=O 49146,CCCC(O)C(=O)N1CCC(C)(NC(=O)Cc2nc(C)sc2C)C1 49147,c1(C(=O)NCC2CC(CNC(=O)COC3CCOCC3)C2)ccc2ccoc2c1 49148,Cn1nnc2c1CCN(N1CCC3C(CCCN3C(=O)OC(C)(C)C)C1)C2 49149,CCC(CC)(CC)C(=O)N1Cc2occ(C(=O)NCC3CC(F)(F)CO3)c2C1 49150,CC1(C)C(NC(C2(CO)CCOCC2)=O)CC1CNC(=O)Cc1cncnc1 49151,C1(NC(CCn2c(C)ncc2)=O)CC2CC(C1)N(C(=O)C(=O)NC(C)C)C2 49152,N1(C(c2cc(C)on2)C(=O)NC2CC2)C(CN(C)C)CC2CC12 49153,C(=O)(C1=CCC2CCC1N2C(c1n[nH]c2ccccc12)=O)NCCCC(C)CO 49154,C1(CNC(CCCCOCC)=O)N(C(=O)C=C2CCC(C)CC2)CCCC1(C)C 49155,C12(CNC(c3ccc(OC)nc3)=O)CCCN(C(=O)CCc3nccs3)C1C2 49156,C(=O)(C(O)CC(C)(C)C)N(CC(C)O)CCNC(=O)Cc1nccn1C 49157,C12(CC(=O)NCCSCC=C)CCC1CN(C(C1(OC)CC(C)(C)C1)=O)C2 49158,CCC(C)C(O)C(C)C(=O)N1CCN(CCNC(c2ccc([N+](=O)[O-])o2)=O)CC1 49159,C#Cc1cnn(CC(N2CCC(NC(=O)CCc3cc(C)on3)C2CC)=O)c1 49160,C(CC(C)N(C)CCOCCCCC)OCCOC 49161,C=C(C)C(CC(=O)N1CCCCC1CNC(c1csnc1C(=O)OC)=O)OCC 49162,C(=O)(C(C(C)C)NS(N)(=O)=O)N1CCC(C(C)(C)NC(C(CSC)O)=O)C1 49163,Cc1cncc(NC(C23CC(OCC(=O)NC4CCCC4C(C)(C)C)(C2)C3)=O)c1 49164,O=C(CC1CC(NC(c2ccc([N+](=O)[O-])cc2)=O)C1)N=c1cc(C2CC2)[nH][nH]1 49165,C(=O)(C(C)C(C)(F)F)N1CCCC(CN2CCN(C(C(C)NC(N)=O)=O)CC2)C1 49166,C(=O)(C1CCc2ccccc21)NC(C(C)(C)NC(Cc1c(C)con1)=O)C 49167,C1(N(C(=O)CC2(C)CCC2)CC)CCCN(C(C2(C)CCCOC2)=O)C1 49168,C1(C(=O)NCc2c(C(=O)NC3(C(C)(F)F)CCC3)c[nH]n2)CCNC(=O)C1 49169,c1(CCC)cc(C)c(NCCOc2cccc(C(C)C)c2)cn1 49170,N1(C(=O)CCOC2CCC2)CC2(CC2)CC1CNC(C1(CC2CC2)CCC1)=O 49171,Cc1cccnc1C=CC(=O)NCC(C)CN(C(=O)CN1CCC(F)CC1)C 49172,CS(=O)c1ccc(C(N2CCC(C)(C)C2CNC(=O)Cc2nc[nH]n2)=O)cc1 49173,C1(O)(CCNC(C=C(C)C)=O)CCCN(C(=O)C=Cc2cnc(C(C)(C)C)s2)C1 49174,C(=O)(C1COc2ccc(Cl)cc21)NC1C=CCN(C(CCc2c[nH]c(=N)[nH]2)=O)C1 49175,CC(C)(CC(=O)N1CCCC1C1CCN(C(c2snnc2C2CC2)=O)C1)C(F)F 49176,c1(OC)ccc(C2(C(=O)NCC3(NC(=O)C(C)OC)CCC3)CCC2)cc1 49177,C(C1=NOC2(CCC2)C1)NC(C(C(C)CN(C(=O)C(=O)NCC1CC1)C)F)=O 49178,c1(CCC(=O)NC(C2CCCN2C(c2cnc[nH]c2=N)=O)(C)C)ccc(Cl)nc1 49179,C1(C(=O)NC(C(=O)NCCCCC)CC2CC2)CC(N=[N+]=[N-])C1 49180,NS(=O)(=O)CCCC(=O)NCC1CCCCN(C(C2CCCCO2)=O)C1 49181,N1(C(C(CC)F)=O)CCOC(CN(C)C(c2csc(-c3ccsc3)n2)=O)C1 49182,C(C1=CCN(C(c2cc3ccsc3[nH]2)=O)CC1)NC(c1cncc(OC)c1)=O 49183,C(=O)(C(C)(C)C(=O)N1CC2(NC(c3nnc(O)cc3O)=O)CCC1C2)OC 49184,C(F)(F)(C(=O)NOCc1ccccn1)C12CCC(OCC)(C1)C2 49185,CN1CC=C(CC(=O)NC2CC(C3CCN(C(=O)CC4(O)CCCC4)C3)C2)CC1 49186,C(N=c1[nH]cnc2c(Br)cccc12)C12C(CN(C(c3ccc(C)c(F)c3)=O)C1)C2 49187,C1(NC(C2CCC=CCCC2)=O)CCCOC12CCN(C(c1cnoc1)=O)CC2 49188,n1(CC(=O)NC2CCC(CNC(CC3CC(CC)C3)=O)CC2)ccc(O)nc1=O 49189,C(C)(C)(CCC(=O)NCC(O)C(N1CCCC(CCOC)C1)=O)OC 49190,N1(C(CN(C2CCN(C(C)C)C2)C)=O)CCN(C(=O)CC2CC2)CC1CO 49191,C1(C(=O)NCCC(CC)CO)CN(C(C2CC(C)CCO2)=O)CC(C)(C)C1 49192,c1(NC(C2N(Cc3cccc(C)n3)CCC2O)=O)ccc(C(F)(F)F)c(Cl)c1 49193,Cc1c(-c2nc(NS(=O)(=O)c3cccc(Cl)c3)cs2)cccc1[N+](=O)[O-] 49194,C1(NC(COc2cc(C)on2)=O)CN(C(=O)CC2CC3(CCC3)C2)CCC1O 49195,O=S(=O)(c1[nH]c(=NCC2CC2C2CCC2)ccc1Br)N1Cc2cccc(Cl)c2C1 49196,c1(C(=O)NC2C(C)N(C(=O)C(C)C(F)F)CC2)cc(S(=O)(=O)N(C)C)c[nH]1 49197,CC(C)C(C(=O)NCc1cnn(C(C)C)c1)c1ccnc(N(C)C)c1 49198,Cc1nccnc1N1CCN(c2nnc(C3CCOC3)n2CC2CC2)CC1 49199,C(C(CC(F)(F)F)NC(c1cncnc1CC)=O)NC(CSCC#C)=O 49200,C1(NC(=O)C2=CCCC2)CC(O)CN(C(C2CC(O)(c3ccccc3)C2)=O)C1 49201,CC(C)(C)C(CCc1ccc(F)cc1)C(=O)N1CCNC2(CC2)C1 49202,C(=O)(C(C)(C)CC1CC1)NC1C(CNC(C(C)NC(CC)=O)=O)CC1 49203,C1(NC(C2C(C)C2(F)F)=O)CCCN(C(c2csc(-c3ccco3)n2)=O)C1 49204,N1(C(C(C=C)(C)CC)=O)CCC(NC(=O)C2=CS(=O)(=O)CCC2)C(F)(F)CC1 49205,c1(-c2cn(CCCN(C(=O)C(c3cccnc3F)(C)C)C)nn2)cnccc1Cl 49206,c1(C(=O)NCCCC(C)NC(C2N(C(C)=O)CSC2)=O)cc2ncccc2o1 49207,c1(C(=O)NC2CN(C(c3cc(CC)c(CC)o3)=O)C2)c(N)ccc(F)c1F 49208,N1(C(C=CCC)=O)CC2CC(NC(c3cn(C)nc3-c3cccnc3)=O)C1C2 49209,C(C)(c1cccnc1)=CC(=O)NCCN(C(C1(C)CC=CCO1)=O)CC 49210,C=CCC(CC(=O)N1CCSC(C)(C)C1)NC(C1CC2(CCO1)CC2)=O 49211,CCN=c1[nH]cc(C(=O)NC2CN(C(c3cc(C(F)(F)F)cs3)=O)C(C)(C)C2)s1 49212,C1(C(=O)NC(c2ncnn2C)C)CCN(C(=O)CN2CCSCC2)C(C)(C)C1 49213,CSC1=C(C(=O)N2CCN(C(=O)CCC#N)CC2C2CC2)CCCC1 49214,C1(CC(=O)N(C2CN(C(=O)COc3ccn(C)n3)C2)C)CCCC(C)O1 49215,N1(C(CCCCOCCCN=[N+]=[N-])=O)CCC2(CCC2)C(CNC2C=CCC2)C1 49216,N1(C(C(C(C)(C)C)(C)C)=O)CCC(NC(c2ccc(N)cc2O)=O)C(F)(F)CC1 49217,c1(C(=O)NCCC(C)(C)NC(c2cc(OC)no2)=O)ncccc1SC 49218,N1(C(CN(C2CCC2)C)=O)CCN(C(c2nncs2)=O)CC1c1nccn1C 49219,C1(OC)CC(CCN(C)C)N(C(C2CCN(c3ccncc3)C2)=O)C1 49220,c1(-c2cn(CCOCC)nn2)cc(OC)c(Cl)cc1OC 49221,C(CCCC(=O)NC12CCC1CN(C(=O)CC(C)(C)C1CC1)C2)(OC)OC 49222,N1(C(C2(C)C=CCC2)=O)CC2=C(C1)CN(C(=O)CCSCc1ccccc1)C2 49223,N1(C(c2ncn(C)n2)=O)CC(F)CC1CNC(=O)CC1CCC2CC12 49224,c1(C(N2CCC(NC(NCCC=C)=NC)CC2)=O)ncc(C2CC2)cc1F 49225,c1(Cn2cc(C3CCN(C(c4nc(CCC)oc4)=O)C3)nn2)cc(F)cc(Cl)c1 49226,c1(CC(=O)NCC2CCN(C(C=CS(C)=O)=O)CC2)cc2ccccc2s1 49227,c1(OC)ccc(CNC(C(C)C)C(C)(C)O)c2cccnc12 49228,c1(C(=O)NCC(CN(C(C(C)(C)OC)=O)C)C)cccc2nn(C)nc12 49229,N1(C(C2(OC)CC2)=O)CCC2(CC1)CCN(C(c1c(C)ccnc1Cl)=O)CC2 49230,n1(CC(=O)NCC(CNC(CC(C)c2ccco2)=O)O)cnc([N+](=O)[O-])c1 49231,c1(CC(=O)NCC2(CC)CCOC2)ccc(NC(=O)C(C)CC2CCCC2)cc1 49232,Cc1nc2cccc(C(=O)NCC34CCCC3CCN4C(c3cnsn3)=O)c2[nH]1 49233,N1(C(C2CC(CC)C2)=O)CCCC(O)(CN(C(=O)CCC(C)C)C)C1 49234,C1(NC(CC(=O)OCC)=O)CN(C(C2CC(=O)NC2(C)C)=O)CC2(CCC2)C1 49235,c1(C(N(C)CCn2cc(CCS(C)(=O)=O)nn2)=O)cc(F)ccc1C1CC1 49236,[N-]=[N+]=NC1COCC1NC(C1CN(C(=O)CN2CC3CC3C2)CC12CC2)=O 49237,N1(Cc2cc(OC)cc(Cl)c2)C(=O)C2C(C)CCCN2C1=O 49238,C1(NC(CCc2cnc(C)s2)=O)CN(C(=O)C(C)Sc2ccccn2)CC1(F)F 49239,c1(C(N2C3C(NC(C4CCN(CC#C)CC4)=O)C(C3)C2)=O)c(C)ncnc1O 49240,c1(C(=O)NCC2CCCN(C(c3c(OC)ccs3)=O)C2)ccc([N+](=O)[O-])c(F)c1 49241,c1(NC(C2CCN2C(=O)C(c2ccccc2)=O)=O)c(Cl)ccnc1Cl 49242,N1(C(=O)Cc2c(F)cccc2Cl)CC2CCC(C1)N(C(c1ccns1)=O)C2 49243,C1(NC(Cc2cccc(C)c2F)=O)CC2CCC1CN2C(=O)CCC(C)(F)F 49244,Cc1cc(Cl)c(C(=O)NCc2ccc(CNC(=O)CC3CC3(C)C)cc2)s1 49245,CCCC(C#N)C(=O)NC(c1cnn(C)c1)C(=O)NCC(C)CCC 49246,N1(C(CC(n2c(CC)ncc2)C)=O)CC2(CC(NC(C3CCOC3C)=O)C2)C1 49247,C1(F)(CNC(c2cc(C)c(O)nc2)=O)COCCN(C(=O)CS(C)(=O)=O)C1 49248,c1(C(N2C(CNC(=O)C3=CCCC3)CC(C(F)(F)F)C2)=O)ccc2ccnn2c1 49249,CC1CCC(C)(C(=O)NC2CC3(C2)CN(C(c2cc(C(F)F)no2)=O)C3)C1(C)C 49250,Cc1cc(F)cnc1C(=O)NC1(CO)CCN(C(C2(N(C)C)CC2)=O)CC1 49251,C(=O)(C(C(C)(C)O)NC(C1CCCN(C)C1)=O)NCCC1C(C)C1 49252,C(=O)(CCCC(F)(F)F)N1C(CCC)CN(C(=O)COC2CCCC2)CC1 49253,CCCC(CC(=O)N(C)CC1(N(C)C)CCC1)NC(c1cc(Cl)c[nH]1)=O 49254,N1(C(C(C2CC2)OCC)=O)CCC2(CCC(NC(=O)CCc3ccoc3)CC2)C1 49255,c1(C(N(CCC(=O)N(CCOC)C)C2CCC2)=O)ccnc(C)n1 49256,N1(C(C(C)(C)CF)=O)CC2(CCN(C(=O)CCCC3CCCCC3)C2)C1 49257,N1(C(C=C(C)C)=O)CCOC(C)(CNC(=O)C(O)Cc2cnc[nH]2)C1 49258,C1(NC(=O)Cc2cccs2)CN(C(c2coc(C(F)F)n2)=O)C2(CCCCC2)C1 49259,c1(N)ccc(C#N)cc1O.CC(C(=O)NC)OC(C)(C)C.C12CC(C1)NC2=O 49260,c1(C(N(C(CNC(CCCCSC)=O)C)C)=O)cc(N)c(F)cc1C 49261,C12(NC(c3c(C)csc3)=O)CCC(CN(C(=O)CN3CCCCC3=O)C1)C2 49262,C1(C(N(CC(CC)OC)CC)=O)CCN(C(=O)CC2CCCO2)O1 49263,C(=O)(C(C(C)(C)C)OC)N1CC(NC(CN(C)CC)=O)C(c2ccnn2C)C1 49264,N1(C(C=CC(C)NC(=O)C(F)CC2CCOC2)=O)CCCCCC1 49265,CCC(C)(C)CCNC(=O)CC(CNC(C1CCCS1)=O)C1CCC1 49266,C(=O)(C1CCc2nccn21)N1CCN(C(CC2C(C)(C)COC2)=O)CC1CCO 49267,c1(OCN2C(COC)CN(C(=O)OC(C)(C)C)CC2)c(Cl)ccc(F)c1Cl 49268,CC1CC(C)OC1C(=O)NC(C)CCNC(c1ccsc1C(F)(F)F)=O 49269,C(CC(C(=O)NCC1CC(NC(=O)C=CCF)C1)NC(=O)OC(C)(C)C)=CC 49270,c1(C2(C(C)NC(C3CCN(C(COCCC=C)=O)C3)=O)CC2)cccc(F)c1C 49271,C1(CC(=O)NCC2N(C(c3c(C)nn(C)c3Cl)=O)CCC2)CCC2(CCC2)CO1 49272,C(C(CNC(=O)Cc1ccn(C(F)F)n1)CO)NC(CSCCOC)=O 49273,c1(CN(C2CCNCCC2C)C(c2c(C)cccn2)=O)ccc(F)c(Cl)c1 49274,C(=O)(C1CCCc2nn(C)cc21)N1C(=O)CCC1.CC(C)Cn1ccnc1 49275,C(CC(C)(C)C(=O)N1C2CCC(C2)C1CNC(=O)Cn1[nH]cnc1=N)SC 49276,c1(C(=O)NCC2N(C(CC(CCSC)O)=O)CCCC2)[nH]nc2ncnc(O)c12 49277,C1(c2nc(CCCCC)nn2-c2ccc(N(C)C)c(Cl)c2)CCC2CC1C2(C)C 49278,CN1C(=O)CCC1C(=O)NCC1CCCC(CNC(=O)Cc2csc(=N)[nH]2)C1 49279,C1(NC(C(C)(F)F)=O)CC2CC(NC(c3ccn(-c4cncc(F)c4)n3)=O)C1C2 49280,N1(C(C2CC=C(C)CC2)=O)CC2(C(N3Cc4c[nH]nc4C3)=O)CCC1CC2 49281,C(=O)(CCCCCNC(C1CN(C(N)=O)C1)=O)N1CC=C(C)CC1 49282,c1(C(=O)NC(C)CN2CCN(C(c3cccnc3S)=O)CC2)nnc(O)cc1O 49283,C(C(=O)N1CC(CO)(NC(=O)CCCCN2CCCC2)C1)(C(C)C)SC 49284,C1(NC(=O)C=CC=C(Cl)Cl)CCC(NC(=O)CC(=O)Nc2ccc(Cl)cc2)CC1 49285,N1(C(C2C(=C)CC2)=O)CCCC(C2CN(C(c3nc[nH]c3C(C)(C)C)=O)C2)C1 49286,C1(NC(C2N(C(=O)OC)CCC2)=O)CCCCC1NC(C1(C)CCSCC1)=O 49287,c1(SCCC)ccc(C(N2CCC(C)(CNC(C3(C#N)CC3)=O)C2)=O)cc1 49288,C(=O)(C1=CC(O)CCC1)NC1CC2(CN(C(c3c(CC)n(C)nn3)=O)C2)C1 49289,Cc1csc2c(N3CC4CN(Cc5cc(Cl)cc(Cl)c5O)C4C3)ncnc12 49290,c1(C(N2CCN(C(c3cccc(F)c3)=O)C3C2C3)=O)cccc([N+](=O)[O-])c1Cl 49291,C1(NC(c2cn(CC)nc2C2CC2)=O)CCN(C(=O)Cc2ccns2)CC1C 49292,N1(CC(N2CCC(NC(C=CC(CC)C)=O)C(O)C2)=O)Cc2ccccc2C1 49293,c1(CC(=O)N(C2CCN(C(C3CCCOC3)=O)CC2)CC)cccc(SC)c1 49294,c1(NC(C(C=C)O)=O)cccc(NC(=O)NC(C)C)c1 49295,N1(C(CC2(C)CCC2)=O)CCC2CN(C(=O)CSc3ccc(F)cc3)CCC12 49296,N1(C(C(C)OCCCC)=O)CC(C2CC2)(C(=O)N(C)CC2(CO)CC2)C1 49297,c1(C(=O)NC2CCCC(N(C(Cc3cnc(C)o3)=O)C)C2)cc2c[nH]cnc-2n1 49298,Cc1c(C(N2CCC(C(=O)NCCc3noc(=O)n3C)(C(C)C)C2)=O)nnn1C 49299,Cc1cc(C(=O)NC(C)CCNC(=O)C2=CCCC2)cc(Cl)c1 49300,c1(C(=O)NC)ccc(C(=O)NC2CC2C(=O)Nc2cccc(F)c2)cc1 49301,C(=O)(C(C)(C)C1=CCSCC1)N(CC(C)(C)CNC(=O)CCC#N)C 49302,C(=O)(C(C)(C)S(=O)(=O)C1CC1)N1CC2C(NC(C(C)CC(F)F)=O)CC(CC2)C1 49303,c1(C(=O)NCc2cccc(F)c2)ccc(F)c(S(=O)(=O)N2CCC2)c1 49304,N1(C(C=C(CC)CC)=O)CC2CC(NC(c3ccnnc3S)=O)CC2C1 49305,C1(C(=O)NC2(CC=C)CN(C(C3(C(C)(F)F)CC3)=O)C2)CCCCC1C1CC1 49306,Cc1nn(C)c(=O)c(C(=O)NCCCC(C)NC(c2csc(Cl)c2)=O)c1C 49307,CC1CC(CCNC(c2ncoc2-c2ccco2)=O)CCN1C(=O)COCCF 49308,C(=O)(C(F)CCC(C)C)NC(CC)CC(=O)NCCCC(C)O 49309,C1(CC)CN(C(=O)C(O)C(C)(C)C)CCC1NC(c1cc(O)ccc1C)=O 49310,N1(C(C(C)=C(CC)C)=O)CCC2(CCN(C(=O)C(C)(C)C(F)F)C2)C1 49311,C1(NC(c2c(C)snc2)=O)CCCC(NC(=O)CC2CCC(C)CC2)C1 49312,C1(C(=O)NC2CC3CC3C2)CCCN(C(C2(CCF)CCC2)=O)CC1 49313,c1(CNC(c2cnc(C)n2C)=O)ccc(CNC(c2c(C)ncn2O)=O)c(F)c1 49314,c1(C(=O)NC2(C)CCN(C(C3CC(C4CC4)=NO3)=O)C2)csc(=NC2CC2)[nH]1 49315,Cc1cc(C(N2CC(NS(=O)(=O)CCCCl)C3(CC3)C2)=O)c(F)cc1Br 49316,CC(C)(C)CCC(N)CNCc1cnccc1Cl 49317,C(=O)(CCCS(C)(=O)=O)NCC1(F)CC(NC(C(c2c(C)cccc2)C)=O)C1 49318,c1(OC)cc(F)ccc1NC(c1ccnc(C)c1N)C 49319,N1(C(CCCO)C(F)(F)F)CCc2cc(Nc3ncccn3)ccc21 49320,CC1=C(C(=O)N2CCC(NC(=O)CC3(O)CCOC3)C(CO)CC2)CCS1(=O)=O 49321,C1(C#N)(C(=O)OCc2cc(C)c(Cl)cc2)CCCCCCC1 49322,c1(CC(=O)NCCOC2CCN(C(CCSC)=O)C2)nn(C)cc1Br 49323,Cc1cn(C)cc1C(=O)NCC(C(=O)N(CCC(=O)NC1CC1)C)N(C)C 49324,N1(C(CCn2c(C)nc(C)n2)=O)CCC2CCN(C(C3CCNC3=O)=O)CC2C1 49325,C1(NC(c2c(CC)nc[nH]2)=O)CCN(C(=O)Cc2cnn(C)n2)C12CCCC2 49326,C(=O)(C1=NN(CCO)C(=O)CC1)N1C(C)C(CC2CC2)CCC1 49327,CC(CC(F)(F)F)C(=O)NC(C)CN(C)C(c1c(O)cc(O)cc1O)=O 49328,N1(C(C2CN(C(C)=O)C2)=O)CC2(NC(c3cncs3)=O)CC1C2 49329,c1(OC)ccc(CC(=O)NC2CCCC2NC(C2CN(C)CCO2)=O)cc1Cl 49330,CCC(C(=O)NCCC1(C(N2CC(C3CC3)(COC)C2)=O)CCCC1)C(C)C 49331,C(C(=O)NOCCC1CC1)(N(C(C(C)SC(C)(C)C)=O)C)C1CC1 49332,c1(C(=O)NCCc2ccc(CNC(C)=O)cc2)onc(C)c1-c1ccccc1 49333,C(=O)(CC(C)(C)C(F)F)N1CC(F)CC(NC(C(C)S(N)(=O)=O)=O)C1 49334,CN1CCN(C(c2cc3occc3s2)=O)C(CNC(c2ccc(O)c(O)c2)=O)C1 49335,Cc1nc(O)[nH]c1C(=O)NCC1CC1CNC(c1csc(C2CCCCC2)n1)=O 49336,N1(C2CCN(C(C(C)=CC)=O)CC2)CCN(C(C2CCC3(CCC3)O2)=O)CC1=O 49337,C#CCCCCCCC(=O)NC1CC(F)CN(C(=O)C(c2ccc(C)o2)C)C1 49338,N1(C(C(C)NC(COC)=O)=O)CC2CCC(C1)C2NC(=O)CC1CC=CCC1 49339,c1(C(=O)NCC2(C)CCN(C(C3(OC)CC3)=O)C2)c(C)nn(C)c1OC 49340,c1(CN2CCC(C(=O)Nc3cc(C(=O)OC)cc(Cl)c3)C2)c(F)cc(O)cc1F 49341,Cc1cnn(CC(=O)NC2C=CCN(C(C3CCCCC(=O)N3)=O)C2)c(=O)c1 49342,c1(NC(C(C)(N(C)C(c2ccnnc2)=O)C2CC2)=O)ccc(O)c(=O)cc1 49343,c1(C(=O)NC2CN(C(C(C=CC)O)=O)CC2O)cnc2c(c1)COCC2 49344,C(CC(=O)N1CC2CC2(CO)C1)(C(F)F)NC(CC1C=NN(C)C1=O)=O 49345,C1(O)(C(C(=O)NC(c2ccc(C)s2)C)NC(c2cc(CC)on2)=O)CCCCC1 49346,c1(CC)cc(C(=O)N(CC(C)(C)C(=O)NC(CO)C(=O)OC)C)nn1C 49347,C(C)(CCC(=O)N1CC(O)(CNC(C2CC(=O)N(C(C)C)C2)=O)C1)SC 49348,C(=O)(CC(C)P(C)(C)=O)N(CC(C)(C)NC(C=C(C)c1ccsc1)=O)C 49349,C1(CC(=O)NCCOCCNC(C(C)NC(CC)=O)=O)C(=O)NN=C1C 49350,C(=O)(C(C)C(F)(F)F)NCCN(C(=O)C(C)COC)CCC 49351,c1(C(=O)NC(=O)CN(C2CCC(C(C)(C)C)CC2)C2CC2)ccc2nn[nH]c2c1O 49352,C1(C(C)C)CN(C(c2cnc(O)c(Cl)c2)=O)CCN1S(=O)(=O)C1CC1 49353,N1(CCNC(C(N(C(=O)CCCC2CCCO2)C)C2CC2)=O)CCCOC1=O 49354,C(=O)(CC(CC(C)C)NC(C1CCC(C)=C(C)C1)=O)NCC(C)(C)OC 49355,C1(C(=O)NC23C(CN(C(c4cc(C)[nH]n4)=O)C2)C3)CCc2ccc(F)cc2C1 49356,c1(C(=O)NC(CC)CNC(c2csnn2)=O)cc(N)c(N)cc1F 49357,N1(C(CCN(CCCCC)C)=O)CCN(C(C2CC2OC)=O)CC1C1CCC1 49358,c1(OC)ccc(CC(N2CCC(CNC(C34CCC(CO3)C4)=O)C2)=O)nc1 49359,c1(C(N2C(COC)CN(C(=O)C=C3CCC(C)C3)CC2)=O)cc(S(C)(=O)=O)co1 49360,C1(COC)CN(C(=O)CC2CCCC2)CCN1C(C1CCCC(=O)N1C)=O 49361,C12(NC(c3ncn(CC)c3)=O)CCCC(NC(c3ccsc3C)=O)(C1)C2 49362,c1(C(=O)NCC2(NC(COCC)=O)CC3CCC2C3)ccc2snnc2c1 49363,C12(C(=O)NCCCc3ncco3)CCC(CC1)N(C(=O)C=CC1CCOC1)C2 49364,C(=O)(CCCS(=O)(=O)NCC1CC1)N1CCN(C(CNC=O)=O)C(C2CC2)C1 49365,S(=O)(=O)(CC(=O)NC1CCCC1(C)CCN1CCC(COC)CC1)N(CC)CC 49366,C1(C(=O)OCC)CC(n2ccnn2)CN1S(=O)(=O)CCC1CC1 49367,c1(OC)cccc(C=CC(=O)NC(C)CC(C)NC(c2ccc(C)nc2C)=O)c1 49368,c1(C(=O)NC2CC(CC(=O)NC(C=C)(C)C)C2)cn(C)nc1SC 49369,c1(C(=O)NCCCCNC(C2C(C(=O)NCC#C)C2)=O)cccc(C(N)=O)c1F 49370,c1(CC)nc(C(=O)NCC2COCC2NC(=O)Cn2cc(Cl)cn2)co1 49371,C1(NC(c2ccc(F)o2)=O)CCC12CCN(C(c1ccc(F)c(F)c1F)=O)CC2 49372,c1(NC(C2(NC(CC3CCC(C#N)C3)=O)CC2)=O)cccc([N+](=O)[O-])c1 49373,c1(C(N(CC(C)NC(=O)CNC(=O)C(F)(F)F)C)=O)nc2ccccc2cc1Cl 49374,C1(C2(O)CN(C(C3CCCC3(F)F)=O)C2)(CNC(C=C(CC)C)=O)CC1 49375,C1(C(=O)NC(CNC(CCC)=O)C2CCC2)CCCN1C(c1ccncc1)=O 49376,c1(N)nnn(CCC2CCC2CN(CC=C)CC2(c3sccc3C)CC2)c1C 49377,C1(NC(c2cncc(OC)c2)=O)CCN(C(=O)COc2cccc(Cl)c2)CC1F 49378,C1(C(N(C2CCNCC2)C)=O)C=CCCN1C(C1(c2ccccn2)CC1)=O 49379,N1(Cc2ccn(CCC)c2)CC2C(CC1c1nc(C(=O)N(C)C)no1)C2 49380,c1(C(=O)NCC2(C)CN(C(C(C)O)=O)C2)cc(C(C)(C)C)ccn1 49381,C(N=c1[nH]ccn2cnnc12)c1cc(OC)c(Br)cc1 49382,C1(CNC(c2coc(Cl)n2)=O)CCN(C(c2cnc3ccnn3c2)=O)CC1(F)F 49383,C=Cc1cnn(C)c1C(N1CC2CC1CC2NC(=O)C(=O)C(C)(C)C)=O 49384,CC1CC(CNC(=O)C=CC(=O)NC(c2ccco2)=O)CN1C(c1ccc(CO)o1)=O 49385,Cc1ccc2c(c1C)OCCC2NC(=O)NC1(C)CCC(=O)N1C 49386,C1(C(=O)NCCC2C(C)C2)CN(C(=O)CC2CCOC2=O)CC12CC2 49387,n1(-c2cccc(C)n2)nc(-c2ccc(CN)nc2)nc1C1CCCn2ccnc21 49388,c1(SC)ccc2cc(C(=O)NCC(C(C)C)NC(=O)C(CO)NC(N)=O)[nH]c2c1 49389,C1(C(=O)OC)CC(F)(F)CCN1C(=O)OC(C)(C)C.C1(OC)CCN2C1C2=O 49390,C#CCC(C(=O)N(CC(C)N(C(=O)Cc1csc(Cl)n1)C)C)C1CC1 49391,N1(C(c2cc(C)oc2)=O)CCC2(NC(c3cc(CC(C)C)c[nH]3)=O)CCCC12 49392,c12nocc1C(=O)NC2.C(C(F)CO)NC(C1(CC(C)=O)CC1)=O 49393,c1(C(=O)OCC(=O)NC2CCN(C(C)=O)CC2)[nH]c2ccc(C(=O)O)cc2c1C 49394,C1(C(N(C)Cc2ccoc2)=O)CC(NC(c2nc[nH]n2)=O)CCO1 49395,N1(C(C2(F)C(C)C2)=O)CCC2(CCC2CNC(c2ccco2)=O)CC1 49396,CC(C)CC(=O)NCC1CCN(C(C2CNC(=O)N2)=O)C1 49397,CC(C)CCCOCC(=O)N(CCCN(C)C)CCNC(C1CC1Br)=O 49398,C1(OC)CCC12CC(C(=O)NCC13CC(CO1)N(C(=O)C(C)(O)C1CCC1)C3)C2 49399,c1(CNCC2CC3(CC(NC(CCSCC(N)=O)=O)C3)C2)cnc2n1CCCC2 49400,CC(C)(C(=O)N1CC(n2cc(CNC(=O)C(O)(C3CC3)C3CC3)nn2)C1)C1CC1 49401,c1(CCC(=O)NCC2CCN(C(C3CNC(=O)N3)=O)C23CC3)ccc(Cl)c(Cl)c1 49402,Cn1nc(CC(=O)NC(C)(CNC(C2CC23CCC3)=O)CO)cc1C(F)(F)F 49403,c1(OC(C)CNC(=O)NCc2nc(-c3ccccn3)no2)ccccc1Br 49404,N1(C(C(n2c(C)ncc2)C)=O)CC2CCC2(CCNC(c2cc(Cl)n(C)n2)=O)C1 49405,c1(C(=O)NC(CNC(c2c(C)cno2)=O)C(C)(C)C)c(Cl)ccc2ccoc12 49406,C1(C)(C(=O)NCc2ccc(C(N(C)Cc3n(CC)ccn3)=O)s2)CCOC1C 49407,c1(CC(=O)NCCCCCNC(=O)CC2(O)CC2)ccc2n[nH]cc2c1 49408,c1(C(c2nnnn2C(c2cccs2)C2CC2)NC(C(C)(C)OC)C)cnc(Cl)n1C 49409,n1(CC)nncc1C(=O)NCC(O)C(=O)NCC(C)N(C)C 49410,N1(C(C(C)OCC)=O)CC(C)(C)CCC1CNC(c1cn(CC(F)(F)F)cn1)=O 49411,C1(CNC(C#CC2(CC)CC2)=O)CCC(C)(C)CN1C(c1csc(C2CC2)n1)=O 49412,C=CCC(C(=O)NC1CCSC12CN(C(c1ccc(Cl)o1)=O)C2)C(C)C 49413,N1(C(C(CCC)N(C)C)=O)CC(NC(c2cccc(C(=O)OC)n2)=O)C(C)(C)C1 49414,C1(c2c(CC)cccc2)CCCN(C23CC(C)(C2)C3)CC1 49415,n1(C(C)C)nnnc1C(C1CCCC1)NC(c1cccnc1)c1ncsn1 49416,C(=O)(C(C)(C)CCCF)N(CCCCCNC(C(C(C)C)OCC)=O)C 49417,CC12CCC(C(=O)NCC(O)CNC(=O)C(C)(C)n3cc(Br)cn3)(CC1)CO2 49418,C1(NC(CCCc2[nH]c(=N)sc2)=O)C2CN(C(c3ccc(CC4CC4)s3)=O)CC12 49419,N1(C(c2ccn(CCOC)n2)=O)CCC2CN(C(C3CC4(CC4)CO3)=O)C2C1 49420,C1(C(N2C(C(C)O)CC2)=O)CCN(C(C2(C)CNC(=O)C2)=O)CC1(C)C 49421,c1(C(N2CCN(c3c(Br)cnc(C)n3)CC2C)=O)ccc(Br)c2ccccc12 49422,c1(SC)ccccc1C(N1CCOC(CCCNC(C2CCCN2C=O)=O)C1)=O 49423,N1(C(=O)CC2CC(F)(F)C2)CCCC1C1CCCN1C(C1SCCCS1)=O 49424,C1(CC(=O)NC(CCNC(C(C)O)=O)C)CC(F)(F)C1 49425,C1(CNC(C(C)(C)F)=O)CC2(CCN(C(c3ccc(N)c(Cl)c3)=O)C2)CO1 49426,N1(C(CC(=O)OC(C)(C)C)=O)CCC(NC(C2CC2(F)F)=O)C12CCCC2 49427,CCCC(C)CC(=O)NC1(C(=O)NC2CCCNC2=O)CCOCC1 49428,C(=O)(C(O)C(C)(C)C)NC1(NC(CN(C2CCCC2)C)=O)CCC1 49429,CC1CN(C(C2(C)CCC(=O)C2)=O)CC1NC(=O)CSc1cccc[n+]1[O-] 49430,C(=O)(C1=C(C#N)CCC1)N(C(C)CNC(C1CCCN1N=O)=O)CC 49431,CCC(C)(CO)C(=O)NC(CNC(c1cncc(F)c1)=O)C(C)(C)C 49432,c1(C(N2C3CCC(CNC(C(C)(C)SC)=O)(C3)C2)=O)ccc2c(c1)COC2 49433,c1(NC(=O)CC2CCN(C(=O)Cc3ccc(F)cc3Br)C2)ccc2c(n1)CCC2 49434,N1(C(C(c2ccccc2)=O)=O)CCC12CN(C(c1cc(O)cc(Cl)c1)=O)C2 49435,c1(OC)ccccc1SCNC(=O)C(c1sc(Br)cc1C)N(CC(C)(C)C)C 49436,CP(C)(=O)c1ccc(C(=O)NCC2(F)COCCN(C(=O)CC3CCC3)C2)cc1 49437,C1(N(C(=O)Cn2ncnn2)C)CCC(NC(c2ccnn2CC(F)F)=O)C1 49438,CCCS(=O)(=O)CC(=O)NC(C)CC(C)NC(=O)COc1ccc(Cl)cn1 49439,N1(C(CCNC(=O)NC)=O)CCCN(C(c2cc(C(C)(C)C)ccn2)=O)CC1 49440,C=C(C)c1ccccc1NC(c1cc(CNC(C2C3CC(=O)CC23)=O)no1)=O 49441,N1(C(c2c(CC)cns2)=O)CCOCC(C(N2CC=CC2C(=O)NC)=O)C1 49442,CN1CCCC(CCC(=O)N(C)CCC2CCN(C(C3(O)CCC3)=O)CC2)C1 49443,c1(C(C)NC(C2N(C(CCOC)=O)CC2C)=O)cccc(C)c1 49444,C#Cc1ccc(C(=O)NCCC2CC(NC(c3ccc(C#N)o3)=O)C2)cc1C 49445,C(C(C)CC(=O)N(C1CC1)C1CC1)NC(CC=CCC)=O 49446,c1(C(=O)NC(CN(C)C)C(=O)NC2CCC(C)(C)C2)ccc([N+](=O)[O-])o1 49447,N1(C(c2cc(CC)nn2C)=O)CC(C(=O)NC(CO)C(N)=O)C(C2CC2)C1 49448,C1(C)(C(=O)NCC(CC)NC(c2nocc2Cl)=O)C(C)(C)C1(C)C 49449,Cc1cc(C(N2CC3C(NC(=O)CC4CCC(C)(C)C4)C3C2)=O)n(C)n1 49450,CCC(C(F)(F)F)NC(c1cc(CNC(C2COCC(C)O2)=O)[nH]n1)=O 49451,CC(C)C(C(=O)N1CCC(NC(C2CC3(CC3)C2)=O)C1)n1cc(Br)cn1 49452,c1(-n2c(-c3ccc(C(CC)C)cc3)nc(CC3(C)CC3)n2)ccc(F)c(Cl)c1F 49453,c1(C(N2CC3C(CNC(=O)CNc4ccccc4)(C3)C2)=O)ccc2scnc2c1 49454,c1(OC)ccc(C(=O)NCCC(C)N(C(=O)CC2CCC(=O)N2)C)c(O)c1F 49455,CCC(C)(C)C(C)CC(=O)NCCC(C)NC(c1ccc(OCCOC)nc1)=O 49456,C1(CNC(COC(C)=O)=O)C2CN(C(c3cnn(-c4cccc(Cl)c4)c3)=O)CC12 49457,C1(C(=O)NCc2nc(-c3ccc(C)cc3)oc2)CN(C)CC(C)O1 49458,N#Cc1ccc(C(N2CC(CO)(NC(=O)C=Cc3cscn3)C2)=O)s1 49459,C1(NC(C2(CC(=O)OC)CC2)=O)CC(C(=O)NC2CNC(=O)C2(C)C)=CC1O 49460,c1(CN2CC(NC(C(C)n3ccnc3)=O)C(F)C2)cccc2c1OCC2 49461,C1(C(=O)NC(CNC(=O)CCCC2CCCC2)C2CC2)CCCC(CF)C1 49462,c1(C(=O)NC2(n3cccn3)CC2)cc(O)nc2c1CN(C(C1(F)CC1)=O)CC2 49463,C1(NC(C=NOC)=O)CCC(O)CN(C(=O)CC(C(F)F)n2cccn2)C1 49464,C(=O)(CC(C)CCC)N1CC(CNC(C2N(C(=O)OCC)CSC2)=O)(OC)C1 49465,CCC1CC(=O)NC(C(=O)NCC2CCC2)CN1.n1(C2CC2)ccnn1 49466,C1(C(N2CC(CNC(=O)C=CC3CCCC3)C(C)C2)=O)(OC)CCC(C)CC1 49467,CCCCC(C(=O)NO)NC(=O)NC1CCOCC1F 49468,C1(C(N(C(C)C(F)F)C)=O)CCC2CCCCN2C1 49469,c1(OC)cccc(C(=O)NC(C)C(c2ccc(F)cc2)NC(c2cc[nH]n2)=O)c1 49470,c1(COC)nc(NCC2CC(=O)N(C)C2=O)cc(=NCc2cccs2)[nH]1 49471,c12ccnc(c1)CC(=O)N1CCC1CNC2=O.C1(C(=O)NC)(OC)CC1 49472,S(=O)(=O)(c1ccc(NCC2=CCCC2)c(C#N)c1)NCC1CCCN(C(C)=O)C1 49473,c1(C(COC(Cc2ncn(C)n2)=O)=O)ccc(C(F)(F)F)cc1 49474,c1(C(N2CCC(NC(=O)COC)C2)=O)ccn(CCC2CC2)n1.c1ccccc1 49475,N1(C(c2cc(-c3cccs3)on2)=O)CC2(CCN(C(C3(C(F)(F)F)CC3)=O)C2)C1 49476,C1(C(=O)NCC2CC(NC(CCC3(C)CC3)=O)C(O)C2)Cc2c(F)cccc2O1 49477,C1(NC(C(C)SCCCC)=O)(CNC(=O)CC(C)N(C)C)CCCC1 49478,N1(C(COCCC)=O)CC2(CC1CNC(=O)Cc1cc(C)[nH]n1)CC2(F)F 49479,c1(C(=O)NCC2CC(C(N(C3C4CCCC34)C)=O)C2)cc(C(N)=O)[nH]n1 49480,C1(C2CCCN(C(c3csc(=N)[nH]3)=O)C2)(NC(CCC(=O)NCCC)=O)CC1 49481,C(=O)(CCCCCC)NCC12OCC(CNC(C(C)OCCC=C)=O)(C1)C2 49482,c1(C(=O)NC(CC)CNC(=O)C(C)c2cncs2)ccc(F)cc1OC 49483,C(=O)(CCC(=O)c1cc(C)sc1C)NCCN(C(=O)CC1CCS(=O)(=O)C1)CC 49484,CC(C)CC(N=c1[nH]c(=NC2CC(F)(F)C2)[nH]c2ccc(Cl)cc12)c1cccs1 49485,O=C(CC(C(F)F)NC(C1(F)CC1)=O)NCC1(F)CCOCC1 49486,CN1CCC2C(CCN2C(=O)CCC2(NC(=O)COc3ccccc3)CC2)C1 49487,C1(C(=O)NC2(C(=O)N(CC(=O)NC(C)(C)C)C)CCN(C)C2)CCCC1C1CC1 49488,C(=O)(N1CCC(C(=O)NCC(F)CO)O1)c1nc(=N)[nH]cc1 49489,C1(NC(c2c(CC)ncs2)=O)CN(Cc2ccn(CC(F)(F)F)n2)CCC1C 49490,C1(C2CCC2)(CN2C3CC(C2)NC3=O)CCC1.C1(CC)(CC2CC2COC)CC1 49491,C(=O)(N=c1[nH][nH]c2cccnc12)C1CCC(NC(c2ccccc2O)=O)C1 49492,C(=O)(CCC(F)(F)F)NCC1CC(O)(CNC(c2c(CC)oc(C)c2)=O)C1 49493,C(=O)(C1CCc2ccccc21)N(C1CC2CC1N(C(=O)CS(C)(=O)=O)C2)C 49494,N#Cc1c(C(=O)NCC2(O)CCN(C(=O)C(=O)NCC(F)(F)F)C2)cccc1F 49495,c1(C(N2C(CC(=O)NCC(C)CCCO)CCC2)=O)cn(C)ccc1=O 49496,N1(C(c2c(CC)[nH]cc2)=O)CCC(C)(CNC(C2CCC(CC)O2)=O)C1 49497,Cc1cc(F)c(C(=O)NC(C2CCN(C(=O)CP(C)(C)=O)C2)C)c(Br)c1 49498,c1(OC)ccc(C(CO)N(C)C2CC2)cn1.C12CCCN(C1)C(=O)CNC2=O 49499,C(=O)(CCS(N)(=O)=O)NCC(C)(C)OCC(=O)N(C)Cc1nccn1C 49500,C(=O)(CCCCC(C)(C)C)NCC(C)(CC)NC(CCC(=C)Br)=O 49501,CCCCC(CN(C(=O)C#CCNC(=O)CSCC)C)CC 49502,C1(C(N2CC(C)C(CCNC(=O)CCCCCF)C2)=O)CCc2c[nH]nc2C1 49503,c1(CC)nnc(C)cc1C(=O)NC(C)(CNC(c1cc(C(F)F)[nH]n1)=O)CO 49504,Cc1cc(O)ncc1C(=O)NC1C2CC1N(C(=O)CN1CCC(=O)CC1)C2 49505,Cc1nc2sccn2c1C(=O)NC1CN(C(c2cc[nH]c2)=O)CC1C 49506,C1(C(=O)NC(C)C(=O)NO)CCC(C)(C)N(C(=O)CC2CCCCCC2)C1 49507,C(=O)(CCC(=O)Nc1nccs1)NCC(C)N(C)C(c1cccc(O)c1)=O 49508,N1(C(C(C)CO)=O)CCN(C(=O)CCC2OCCO2)C(CF)C1 49509,c1(C(=O)NC2(C)CC(C(=O)Nc3cnc(OC)nc3)C2)nccc(C)c1F 49510,c1cc(Cl)cc(Cl)c1.N1(C(C=CC)=O)CCC(C)C1CNC(c1cccn1CC)=O 49511,Cn1cc(C(F)=CC(=O)NC2CC(NC(c3conc3C3CCCC3)=O)C2)cn1 49512,C(=O)(C(CC(C)C)C(C)C)NCCC1OCCN(C(CC2(NC(C)=O)CC2)=O)C1 49513,c1(OC)ccc(NC(C2CC23CCN(C(c2cnnc(O)c2)=O)C3)=O)c(CO)c1 49514,c1(C(N2C(CNC(Cn3ncc(C)c3)=O)CC2)=O)cncc2cnccc12 49515,C12(NC(=O)Nc3ccc(OCCO)nc3)CCC(O)(CC1)C2 49516,CCCCCC(F)C(=O)N1CCC(C(=O)NC(C23CCC(CO2)C3)C)(C(C)C)C1 49517,C1(CC)CC(NC(=O)CC(C)(C)NC(C2CC(O)C(F)C2)=O)CCO1 49518,C1(CNC(CNC(C)=O)=O)CN(C(=O)C(C)(C)N(C)C)CC(C)(C)C1 49519,C#CC1CCCN(C(=NCCOCC)NCC(CC2CCC2)CO)C1 49520,C1(SC)CN(C(=O)C(N2CCCC(C)C2)=O)CC1NC(c1cn(C)nn1)=O 49521,C=CC(C)(CC)C(=O)NC1CCCC1NC(c1c(C)coc1-c1ccccc1)=O 49522,N1(C(C(C(=O)OCC)F)=O)CCN(C)C(C(=O)NCC2=CCCC2)C1 49523,c1(OC)ccc(CC(=O)N(C)CC2CN(C(=O)Cc3ccsc3)CCO2)c(F)c1 49524,c1(C(C(=O)NCC2CCCO2)N(CCCC)CC)nc(C2CC2)cs1 49525,C(=O)(NNc1ccc(S(=O)(=O)C(F)F)cc1)c1c(OC)c(F)c(F)c(F)c1 49526,C(CC(C(=O)N(C)C)c1ccccc1)=C(C)C.c12ccc(nc1)NCCNC2=O 49527,C1(C)(C(N2CCC(N(CC#C)C(c3cnc[nH]3)=O)CC2)=O)CCCNC1=O 49528,N1(C(c2ccc(NC(N)=O)cc2)=O)CCC2CCN(C(=O)CC3CC34CC4)CC12 49529,c1(C(=O)NC2CCCN(C(C3(COC)C=CCC3)=O)C2)nccc2ccccc12 49530,C(C)(CCCCNC(=O)C(C)c1cccs1)NC(C1N=C(C)SC1)=O 49531,C1(CNC(C(C)=C2CC2)=O)CC2(CCN(C(c3ccnc(S)c3)=O)CC2)CO1 49532,c1(C(=O)NC(CCOC)CNC(C2(C)CC=CC2)=O)ccc2cnn(C)c2c1 49533,CC1(C(N2CC(NC(=O)CC3(O)CCCCC3)C(CO)C2)=O)CC2CCC1C2 49534,CON(C(=O)C1CCN1C(=O)C(O)Cn1cncn1)C1CCC1 49535,c1(C(=O)OC)cc(OC(C)=O)ccc1Cl.C123CC(C1)(C2)NC(=O)NCC(=O)N3 49536,Cn1ccc2cccc(C(N3CC4CCC(Nc5ncc(O)cn5)C4C3)=O)c12 49537,N1(C(c2cnc(SC)s2)=O)CCN(C(C2CCCC2c2cnn(C)c2)=O)CC1 49538,C1(NC(C2CC(C)SCC2)=O)CCCC2CN(C(=O)Cc3ccn(C)n3)CC12 49539,n1(CC)nc(C(=O)NC2CC(C(N3CC(CO)CC3CO)=O)C2(C)C)cc1O 49540,C(=O)(C(C(C)CC)NC(=O)C(C(CC)CC)OCC)NC1(COCC)CC1 49541,C1(NC(C2(OCC)CCC2)=O)CCN(c2cc(OC)nc(COC)n2)CC1O 49542,c1(SCCC)nc(=NC(=O)N2CCC(OC)C2(C)C)s[nH]1 49543,Cc1ccnc(C(=O)NCC(O)CCNC(C2CCCCCN2C)=O)c1F 49544,Nc1ncccc1C(N1CC2C(CNC(c3cc(=O)cc[nH]3)=O)C2C1)=O 49545,C(=O)(C(O)CC(F)(F)F)N1CCCC(N(C(COCc2ncc(C)o2)=O)C)C1 49546,c1(NC(c2coc(Cl)c2)=O)cccc(NC(C2(C3CCCO3)CCC2)=O)c1 49547,C1(NC(CC(C(=C)C)OCC)=O)COC2(C1)CN(Cc1sccc1Cl)C2 49548,N1(C(C(CC=C)C)=O)C2CCC1CC(C(=O)NC1(C(=O)OC)CC1)C2 49549,c1(C(=O)NC2(CNC(=O)C(=O)NC3CC3)CC2)ccnc2c1CCC2 49550,C1(C(=O)Nc2ccc(C#C)cc2)CN(C(=O)CC2CCCCCC2)CCC1(C)C 49551,C1(C(N2CCC(NC(C3(C(F)(F)F)CCCCC3)=O)CC2)=O)CC12CC(F)(F)C2 49552,CN=c1nc(N2CCC(C(C)COC)CC2)[nH]c(N2CCOCC(C)C2)n1 49553,N1(C(c2c(C(C)C)ocn2)=O)CCCC(NC(=O)C(C)c2ccco2)CCC1 49554,CCC(CC(=O)NC(C1CN(C(=O)C=Cc2ccc(C(F)F)o2)C1)C)OC 49555,C1(CNC(c2ccco2)=O)COCC2(CCN(C(=O)CC3CC4(CC4)C3)CC2)O1 49556,c1(OC)cc(C(=O)NCC2(F)CC(CNC(=O)CN3CCOCC3)C2)ccc1Cl 49557,Cc1cnc(Cl)c(C(=O)N(C)Cc2cccc(CNC(c3sncc3C)=O)c2)c1 49558,N1(C(C2N(C)CCOC2)=O)CC2CCN(C(c3ccc(Cl)c(Cl)c3)=O)C(C2)C1 49559,C(CN=C(NCC(C)C)N1CCC(=C(F)CO)CC1)c1c(OC)ccc(F)c1 49560,C(=O)(CS(=O)(=O)C1CC1)NC1CCCC(NC(=O)COc2cccnc2)CC1 49561,N1(C(CN(S(C)(=O)=O)C)=O)CCC2C(NC(c3sc(F)cc3Cl)=O)CC12 49562,C(=O)(C(C)(F)C(=O)NC(C)C(=O)N(CCC(F)CN=[N+]=[N-])C)OC 49563,c1(SC)cn(C)nc1C(N1CCCC(C(C)NC(C2(O)CCOCC2)=O)C1)=O 49564,N1(C(C2(C)CC(F)(F)C2)=O)CC2CCN(C(C3CC4C=CC3CC4)=O)CCC2C1 49565,N1(C(Cc2cccc(COC)c2)=O)CCC(NC(C2CCCC23CC3)=O)CC1C 49566,c1(CN2CC(C(N3CCC(c4ccccc4)C3)=O)C2)cc(F)ccc1[N+](=O)[O-] 49567,C(=O)(CCCCCN=[N+]=[N-])NCC1CC(CC(=O)N(C2CCCC2)C)C1 49568,Cc1ccc2cc(C(=O)NC3CCCC34CCN(C(C3(CO)CC3)=O)C4)[nH]c2c1 49569,C1(C(N(CC(C)OC)C(C)C)=O)CC(C)(NC(=O)CC2CCOC2)C1 49570,CC(C)(C(=O)NCCc1nnc(O)o1)NC(C12CC(F)(C1)C2)=O 49571,N1(C(COCCOC)=O)CC=CC1CNC(=O)CN1CCC(C)C1 49572,Cc1ccn2ncc(C(=O)NC3CN(C(=O)CC4CC=CCC4)CC3(C)C)c2n1 49573,c1(C(=O)NCC2C(NC(C3C(C(=O)OC)C=C3)=O)C2)n[nH]c2nccc(Cl)c12 49574,CC1CNCCC1C(=O)NCC1CC(C(F)(F)F)CN1C(=O)OC(C)(C)C 49575,N1(C(C(COC)NC(C(COC)OC(F)F)=O)=O)CCN(C)C(=O)C1C 49576,c1(CS(N2C(C(=O)O)CC(=C)C2)(=O)=O)c(SC)cccc1Br 49577,C(CS(=O)(CCO)=NC(=O)c1ccc(-n2ccnc2)cc1)NC(=O)OC(C)(C)C 49578,CC1CN(C(=O)CC(C(F)(F)F)NC(=O)CC(C(Cl)Cl)N(C)C)C12CCOCC2 49579,C12(C(=O)OC)CC(C(=O)NCC3CCC(NC(=O)CCc4ccncn4)C3)(C1)C2 49580,c1(C(N2C(CCNC(=O)C=Cc3cc[nH]n3)CCCC2)=O)cnc2c[nH]nc2c1 49581,C1(n2cc(C#CCNC(=O)CC(O)CF)nn2)CCOC2(CCOCC2)C1 49582,c1(OCCOC)cccc(C(=O)NCCOC)c1.C(=O)(CC(Cl)Cl)N1CCOCC1 49583,N1(C(c2c(CC)ccs2)=O)CCN(C(C2CCN(C)CC2)=O)C(CF)C1 49584,c1(C(N2CC(C)N(C)CC2)=O)c[nH]c2ccc(-c3ccc(OC(F)(F)F)s3)cc12 49585,c1(C(=O)NC2C3(CC(NC(Cc4cnc(C)[nH]4)=O)C3)C2)ccc(N)c([N+](=O)[O-])c1 49586,c1(C(N2C(C(C)(C)NC(C=CS(C)=O)=O)CCC2)=O)cccc([N+](=O)[O-])c1O 49587,C#Cc1ccc(F)c(C(N2CC3CCC2(CNC(=O)Cc2ccsc2)CC3)=O)c1 49588,C1(NCC2CCN(C(C)C)C2)CCCCN1C(c1ccn(CCF)n1)=O 49589,O=C(C#CC1CCCO1)NCC(c1ccc(F)cc1)NC(c1cc(Cl)no1)=O 49590,C1(N(C(C(CC)C)=O)C)CCCCN(C(C2CC=CC2)=O)C1 49591,C12(OC)CC(C(=O)NCC(C)(C)NC(c3cccc(F)c3)=O)C(C1)C2 49592,c1(C(N2CCN(CC(N3CCOCC3)=O)CC2)=O)n[nH]c2c1CCC(F)(F)C2 49593,c1(C(=O)NCc2nc(C(N3CCCC3c3ncc[nH]3)=O)co2)c(O)cccc1Cl 49594,c1(-c2nc(C(C)OC)nn2CC2CCOC2)cc(=O)c2ccccc2o1 49595,c1(OCC)ccc(CN2CCCC(C)(NC(c3nccn3C)=O)C2)cc1OC 49596,C1(NC(C(CCC)OCC)=O)CCN(C(c2cc(C)n(C(C)C)c2)=O)CC1F 49597,N(C1CCOc2ccccc21)(C1C2CCC1CNC2)C(C(CCSC)O)=O 49598,CC1Cn2nc(C(=O)NC(C)CNC(c3cc(C(F)(F)F)n[nH]3)=O)cc2C(=O)N1 49599,c1(CC(C)C(=O)NCC#CCNC(C2CC3(CCCO3)C2)=O)ccc(C#N)cc1 49600,C1(C(N2CC(CNC(C=C(C)C)=O)OCC2)=O)CCN(C)S1(=O)=O 49601,c1(N2CCN(C(c3cc(C)cc(C#N)c3)=O)C3C2C3)ncnc2cccc(F)c12 49602,Cc1cc(Cl)c(Br)cc1C(N1CCCC1C(=O)Nc1nc(C#N)cs1)=O 49603,C=CC1(C(N2CCC(C(F)(F)F)C2)=O)CCN(C(C2CCC2C)=O)C1 49604,N1(C(COCCCC)=O)CC2CCC1C(CNC(=O)CCCc1cnn[nH]1)C2 49605,N1(C(c2ncn(CC)n2)=O)CC(CNC(=O)C=Cc2ccsc2)C2(CCC2)C1 49606,c1(C(N2CC3CCC3(C(N3CCC(O)C3)=O)C2)=O)cccc2ncsc12 49607,C1(CC=C)(NC(C2C=C2C)=O)CCN(C(=O)C(C(C)C)OC)CC1 49608,n1(CC)ccnc1C=CC(=O)NC1CC1CNC(C1COCCO1)=O 49609,c1(OC)ccc(CC(=O)NCC(C2CC2)NC(C2CC3C=CC2O3)=O)c(C)c1 49610,N1(C(c2c(OC)ccc(C)c2)=O)CCC2C(CCN2C(c2cnncc2C)=O)C1 49611,c1(CC)nc(C)c(C(=O)NCC(C2CCCN2C(C2CCCOC2C)=O)(C)C)s1 49612,N1(C(C2(C)CCCCC2)=O)CC(CO)C2(CCN(C(C3COCCO3)=O)CC2)C1 49613,C1(CNC(C2(C)ON=C(C)C2)=O)CN(C(c2c[nH]nc2Cl)=O)C2(CCC2)C1 49614,c1(CC)ccc(O)c(C(=O)N(C(C)CCNC(C2CCC2(C)C)=O)C)c1 49615,C1(CC)C(NC(=O)COc2cccc(C)c2)CCN1C(c1ccsn1)=O 49616,N1(C(c2ccc(C(CC)=O)cc2)=O)CCN(C(=O)C(C)C(C)O)CC1CC(F)F 49617,C1(N(C(C2C(CNC(c3c(CC)non3)=O)OCC2)=O)C)CCC(O)CC1 49618,CCCC(C)(O)C(=O)NCC(C)CNC(=O)CSc1ccc(OC)cc1 49619,N1(C(c2cc(C)c(O)nc2)=O)CCC=C(C(=O)N2CCCCC2C#N)C1 49620,C12(C(=O)NC(COc3cccc(C(=O)OCC)c3)C)CC=CC(C1)OC2 49621,c1(N(C)C)ccc(C(N2CC3C(NC(=O)CN4CC(C)(C)C4)C3C2)=O)cn1 49622,CC1=C(C(=O)NC2(C(N3CCC(C(C)CO)CC3)=O)CCCC2)CCO1 49623,CCCC(CCO)NC(=O)C(CC)NC(=O)C#CC(C)C 49624,C(c1cccc(Cl)c1)=CC(=O)NC(C1CCN(C(c2cc(C)c(C)[nH]2)=O)C1)C 49625,N1(C(C=C(C)Cl)=O)C2CCC1CC(N(C)C(c1ccncc1Br)=O)C2 49626,S(=O)(=O)(c1c(C)noc1C)NCC(=O)NC1C(NC(C(CC)COCC)=O)CC1 49627,c1(OC)c(C(=O)NC(C)C(C)NC(c2cc(-c3ccco3)c[nH]2)=O)csc1Cl 49628,C1(C)(C(=O)NCC2CCN(CCC)C2)CCCN(C(c2cc(Br)nc(Br)c2)=O)C1 49629,C1(CCOC)(NC(=O)CC2(CO)CC2)CCN(C(C2CC2C(C)O)=O)CC1 49630,N1(C(C(COC)N(C)C)=O)CC(CNC(=O)CCn2ccc(C)n2)C2(CC2)C1 49631,c1(CC(N2CCC(CNC(c3ccnn3CCl)=O)C2)=O)cccc(C(F)(F)F)n1 49632,CC(C)C(O)CCNC(C1CC=CCN1C(C1CC2C=CC1O2)=O)=O 49633,C(C(CNC(=O)CC1CCC(=O)N1C)C(F)(F)F)NC(c1c(SC)nn(C)c1)=O 49634,Fc1cccc2nc(N3CCN(CC(F)(F)Cl)CC3)[nH]c(=NCC=C(Cl)Cl)c12 49635,n1(CCOCC)cc(C(=O)NCCNC(C2CCC(C(N)=O)C2)=O)cn1 49636,c1(OCC(N2CCC(N(C)Cc3cccnc3O)C2)=O)cc(F)cc(Cl)c1 49637,CCC(C)C(=O)N(C)CC1(O)CN(C(C2C=C(C)CS2)=O)C1 49638,c1(C(N2CC(NC(C(CCC)O)=O)C(OC)C2)=O)cnc2c(c1)CNC2=O 49639,Cc1ccc(C(F)(F)F)c2c1N(CC1(ON)CC3CCC1CC3)CCC2 49640,c1(NCC2(CO)C(C=C)C2)[nH]c(=NC2CC3(CCCC3)C2)nc2scnc12 49641,CC(C)CCCC(C)NC(=O)CN1CCN(C(C2C=CC=CC=C2)=O)CC1 49642,N1(C(c2c(C)csn2)=O)CCN(C(c2ccc(F)cc2O)=O)C2CCCC2(C)C1 49643,N1(C(C2(COC)C=CCC2)=O)CCCC(NC(c2nnsc2SC)=O)C1 49644,CC1=C(C(=O)NC(CNC(c2ccc(C(C)C)cc2)=O)CC(F)(F)F)CCCO1 49645,N1(C(Cn2c(C)ncc2)=O)C2CCC(C2)C1CNC(C1COC2(CCC2)C1)=O 49646,N1(C(c2ccc(C(C)=O)cc2)=O)CC(C2CCCN(C(=O)C(C)(C)C(C)O)C2)C1 49647,N1(C(c2n(CC#C)cnn2)=O)CCC2C(C(=O)N(CC(=O)NCC)C)C2C1 49648,Cn1ccc(C(N2CC(C)(NC(=O)CC3(O)CCOC3)C2)=O)c1C1CCC1 49649,C1(NC(C2CC2(F)Cl)=O)CCN(C(=O)C(C2CCCC2)C2CCCC2)CC1 49650,N1(C(C2CC(SC)C2)=O)CC2CC2(NC(=O)COCc2cccc(OC)c2)C1 49651,C1(CC(=O)N(C2CC2)CC2C(C)CN2C(=O)OC(C)(C)C)CCC(C)(C)CO1 49652,c1(C(N2CC(NC(C3(OC)CCOC3)=O)C2)=O)cc2c(C)c(Cl)ccc2[nH]1 49653,N1(C(CCC2CC(OC)C2)=O)CCCN(C(c2cc(C#N)ccc2C)=O)CC1C 49654,Cc1cc(NC(c2ccc(S(=O)C(C)C)cc2)=O)cc(S(N)(=O)=O)c1 49655,C1(CNC(c2cn(C(C)C)nn2)=O)(CO)CCCN(C(C2CCCC(F)C2)=O)C1 49656,c1(NC(=O)NCCCCC2CN(C(C3CCCO3)=O)C2)ccc(F)c(F)c1F 49657,c1(C(=O)NC2CC(CNC(Cc3c(C)nsc3)=O)C2)coc2c1CCCC2 49658,C1(C2CCN(C(CC=C)=O)C2)CCCCN1C(=O)CCc1cccnc1 49659,CC1CCN(C(=O)C(N2CCC(C)(c3ccccc3)C2)=O)CC1C 49660,CC1=NOC(C)(C(=O)NCC2CCCN2C(c2cn(CCCF)nn2)=O)C1 49661,C1(CC(N2C(CNC(CSC)=O)COCC2)=O)CN2CCN1CC2 49662,Cc1ccc(N2CC(NC(C3(N4CCCC4)CCCC3)=O)CC2=O)cc1 49663,c1(N2CCN(CCCN(C)C)CC2)nc(N(CC(F)(F)Cl)C)c2ncccc2n1 49664,CC1CC(=O)NCC1C(N1CC(C(C)NC(c2cc(Br)c[nH]2)=O)C1)=O 49665,CC1CC(NC(c2cc(CF)on2)=O)CN(C(c2c[nH]nc2C2CCC2)=O)C1 49666,C12(NC(c3c(C)cc(C)s3)=O)CCOC(CNC(C3CCC(=O)NC3)=O)(C1)C2 49667,CCCC(C)(O)CC(=O)NCC1CC(F)CN1C(=O)Cc1ncc(C)s1 49668,Cc1oc(C(=O)NCCC2(O)CN(C(c3ccc(C(C)C)cn3)=O)C2)cc1CO 49669,C#Cc1ccc(CC(N2CCOC(C)(CNC(c3cnnc(O)c3)=O)C2)=O)cc1 49670,c1(-c2cn(C)c(=O)c(C(=O)NCC3CCS(=O)(=O)CC3)c2)c(F)cc(Cl)cc1F 49671,c1(C(N2CCCC(O)(CNC(CCCOC)=O)C2)=O)cc(OC)cc([N+](=O)[O-])c1 49672,CC1CC(C)(C)CN1C(c1cn(C(C)(C)C)nn1)C(=O)NC1CCCC1 49673,Cc1c(Br)sc(CNCC(=O)CC(C)C)c1Br 49674,c1(C(=O)NCC2(OC)CCN(C(c3ccon3)=O)C2)ccc(F)c(C=O)c1 49675,N1(C(C2(NC(c3n(C=C)ncc3)=O)CCN(C)C2)=O)CCC2(CCC2)C(O)C1 49676,N1(C(C(C)OC(C)C)=O)CCC2C(C1)CN2C(=O)CCCc1ccc(Cl)c(Cl)c1 49677,c1(N2CCCC(NC(C)=O)C2)ncnc(NCC2CCCC2(C)C)c1C 49678,C1(C(=O)NCCC2CCCN2C(c2n[nH]cc2F)=O)CCN(C(=O)C2CC2)CC1 49679,C1(N(C)C(C2CC23CCC3)=O)CC2CC1N(C(c1ccc(N)cc1F)=O)C2 49680,C1(c2nnnn2Cc2ncc(Br)s2)(NCc2sccn2)CC(C2CCC2)C1 49681,N1(C(c2c(SC)ccs2)=O)CCOC2(CCN(C(C3CCOCC3)=O)CC2)C1 49682,C1(NC(=O)Cc2cccc(F)c2Cl)CC12CCC(NC(c1cnsn1)=O)CC2 49683,Cc1cnc(C(N2CCC(C)(C(N3CC(N4CCCC4=O)C3)=O)CC2)=O)c(F)c1 49684,Cc1oc(CN2CCC2C(=O)NC(C)C)cc1CO 49685,CN(CCCC(=O)N(C)CC1CCN(C(C2(C(F)(F)F)CC=CCO2)=O)C1)N=O 49686,c1(C(N2CCC3(C2)CC3(F)F)C(=O)NC2(C)CC2)cnc2ccc(Cl)cn12 49687,C1(COC)(CNC(C2CCCCC2O)=O)CCCN1C(=O)CC1(C)OCCO1 49688,c1(C(=O)NC23CC(NC(CC4CC(C(=O)OC)C4)=O)(C2)C3)ncc(C)cn1 49689,C#CCC(C)(C)C(=O)NCCC1CCC(NC(c2n[nH]cc2OCC)=O)C1 49690,N1(C(c2cc(Cl)c(Br)s2)C(=O)NC)CC2CCCC1C2CNC(=O)OC(C)(C)C 49691,c1(C(N2CCC(CNC(C(CCC)CC)=O)C23CC3)=O)ccc2c(c1)NC(=O)C2 49692,O=C(CCCCCCCO)NC1CC(C(=O)Nc2nnco2)C1 49693,c1(C(=O)NC(C)CCNC(C2(F)CCCC2)=O)cc(Cl)cc(Br)c1N 49694,N1(C(C2CC(OC)C2)=O)CC2CCC(NC(c3c[nH]cc(F)c3=O)=O)CC2C1 49695,C1(NC(C2CCC(C)C2)=O)CN(C(C2C3CCCC23)=O)CCC12CCC2 49696,n1(CC(N2CC(CC(C)NC(C(C=C=C)C)=O)C2)=O)ccc2ccccc2c1=O 49697,C(=O)(CC(C)(C)Cn1cc(CCN2CC(=O)CCC2=O)nn1)N(C(C)C)C1CC1 49698,c1(CCC)onc(C)c1C(=O)NC1CN(C(=O)CCc2ccc(OC)cc2)C1 49699,C1(NC(C=CCOCCOC)=O)COCCN(C(c2cnc(S)n2C)=O)C1 49700,C=C(C)C(CC(=O)NC1CN(c2cc(O)nc(SC)n2)CCC1C)OCC 49701,C12(C(N(C3CCN(C(c4ccc(Br)cn4)=O)CC3)CC)=O)CC(C)(C1)OC2C 49702,c1(CC)cccc(C(=O)N(C(C)CN(C)C(C2(Br)CC2)=O)C)n1 49703,C(CCCC(C)(C)C(=O)NNC(=O)c1csnn1)NC(c1cc(CC)nc(Cl)c1)=O 49704,N1(C(Cc2cnc(C)[nH]2)=O)CC2CCC(C1)C(NC(C1CCC3CC13)=O)C2 49705,CC1CC(C)CN(C(=O)CC2CC(NC(=O)CN3CCCCC3C)C2)C1 49706,C(=O)(C(O)CC(F)F)NC(CC)CNC(=O)Cc1cc(-c2ccccc2Cl)on1 49707,c1(C(=O)NC2C(NC(CC(C)(C)C)=O)CCC2)cc2ccccc2cc1N 49708,c1(C(N(C2CCN(C(C3C4CCCOC34)=O)C2)CC)=O)cccc(OC(F)F)n1 49709,N1(C(CCCCOCC)=O)CCN(C(c2cn(CCO)nc2C)=O)C(C2CC2)C1 49710,C=CCCCC(=O)N1CCC(N2CC(C)(CNC(C34CC(F)(C3)C4)=O)C2=O)CC1 49711,C1(NC(C(C)(C)SC)=O)CCCC(CNC(c2ccc(O)cn2)=O)C1 49712,c1(OC)cnc(F)cc1C(=O)NC1(CNC(c2nnsc2C)=O)CCCCC1C 49713,Cc1ccc2c(C(N3CC(CC(C)NC(C4(S(N)(=O)=O)CC4)=O)C3)=O)coc2c1 49714,C1(C(N(C2(CC(=O)N(CC(COC)(F)F)C)CC2)C)=O)CCCC(C)C1 49715,c1(C(=O)OC)ccc(C(=O)NCC(C2CCC2)NC(=O)C(C)=C(C)C)nc1 49716,C1(C(N(CC)Cc2ccsc2)=O)(CC)CCCN(C(c2ncc(C)cc2F)=O)C1 49717,c1(C(=O)NCC2(CNC(c3c(CC)ocn3)=O)CC2)ccc(F)c(C(C)(C)F)c1 49718,n1(CC(N2CC3C(NC(c4c(C)cns4)=O)(C3)C2)=O)nc2n(c1=O)CCCCC2 49719,C(CC(C)C(=O)N(C1CCC(CNC(c2cc(Cl)cs2)=O)CC1)C)=CC 49720,C1(C(=O)NCCCNC(C2N(S(C)(=O)=O)CCCC2)=O)CCc2nncn2C1 49721,C1(C(=O)OC)CCCN2C1CN(C)CC2=O.c1(CC)ccc(C2CC2)o1 49722,CCC(C)(CNC(=O)C(F)OC(F)(F)F)C(=O)NCC1(CN=[N+]=[N-])CC1 49723,c1(C(=O)NC(c2ccccc2)CNC(c2cn(CC)nn2)=O)cccc(SC)n1 49724,CC12CCC(C(=O)NCCC3CN(C(C4CCCCCC4)=O)C3)(CC1)CO2 49725,c1(CN2C3CN(C(c4c(C)n[nH]c4)=O)CC32)ccc(F)cc1C(=O)O 49726,c1(CC(N2CC(NC(=O)C(F)F)C(F)C2)=O)cc(F)ccc1Br 49727,C1(CC(=O)N(C(c2ccccn2)C)C)CCCN(C(C2CCCO2)=O)CC1 49728,N12CCC(C)C(C1)CNC1CC(C1)CC2=O.C1(C(=O)NCC)(C(=O)OC)CCC1 49729,C1(NC(C(C=C)OC)=O)CC2CCC1(C(=O)Nc1cnc(O)c(C)c1)C2 49730,c1(CC)c(C(=O)NC2CCCC2CNC(=O)Cc2csc(C)c2)csc1C 49731,N1(C(CCN(C)CC)=O)C2CCC1C(C)C(NC(c1nc(C)oc1C)=O)C2 49732,c1(OC(C(=O)N(CC(C)NC(=O)C(C)n2ccnn2)CC)C)ccc(C)cc1 49733,c1(C(N2CC(F)(CNC(c3cc(C(F)F)no3)=O)C2)=O)nccc(F)c1Cl 49734,N1(C(=O)NCc2c(OCCOC)cccc2)CCCC(CO)CC1 49735,C(=O)(C(CN(C)C)NC(=O)Cn1ccnn1)N(C(C(C)SC)C)C 49736,N1(C(C(C)N(C(c2cnc[nH]c2=N)=O)C2CC2)=O)CCSC(C)C1C 49737,c1(CC(=O)NC(C)CC2CN(C(C3CC(C)(O)C3)=O)C2)cc(F)ccc1Br 49738,Cn1cccc1C=CC(=O)NC1(C)CC(NC(=O)CC2CC(=O)NC2=O)C1 49739,O=C(C(O)CC(F)F)Nc1ccc(N2CCCNC2=O)nc1 49740,C1(C(=O)NCCOCCNC(c2nn(CC)nc2C)=O)C2CS(=O)(=O)CC12 49741,N1(C(C(c2ccc(F)cc2)=O)=O)CC(NC(C2CC3C=CC2CC3)=O)CC(O)C1 49742,C1(CNC(C(=O)NC2CC2)=O)CC2(CC(NC(c3cccnc3C(F)F)=O)C2)C1 49743,C(CCCCCNC(=O)CCc1cccnc1Br)N(C(C1C(=C)CC1)=O)C 49744,C(=O)(CCCN(C)N=O)N1CC(CNC(CCC2CC(OC)C2)=O)OCC1 49745,c1(CC)cnccc1C(=O)NC1CC(C(=O)NCC(c2ccccc2)F)C1(C)C 49746,N1(C(C2CCN(C(c3cc(C)c(=N)[nH]c3)=O)C2(C)C)=O)CCC2(CC(F)C2)C1 49747,C=CC(CCC)CC(=O)NC(C(=O)NC1CCCCCC1F)C(C)(C)C 49748,N1(C)CCCC(Cn2cc(C(=O)OCC)cn2)C1.c1c[nH]nc1OC1CCNC1 49749,c1(OC)cc(CN2CCOCC2)c(OC(C)C)cc1I.C12CCCN(C1)C(=O)N2 49750,c1(C(N2CCN(C=O)CC2)C(=O)Nc2ccc(OCF)cc2)cc(Cl)c(Cl)c(Cl)c1 49751,N1(C(c2cc(C)nc(O)n2)=O)CC23CCCC2(C1)CN(C(C1(C)CCCO1)=O)C3 49752,N1(C(c2nc(C(N)=O)sc2)=O)CC2(COC(CNC(c3coc(Cl)n3)=O)C2)C1 49753,NCCCC(O)C(=O)OCC(c1ccccc1)CBr 49754,C(=O)(CC(F)(F)C(C)(F)F)NCCC1(CNC(C2ON=C(C)C2)=O)CC1 49755,N1(C(c2c(CC)cns2)=O)Cc2n[nH]cc2C1C(=O)N1CCC(C)(NC(C)=O)C1 49756,c1(N2CCCCC(CO)C2)nc2c(c(=NCC3CC3(F)F)[nH]1)CSC2 49757,C(=O)(C1=NOC2COCC12)N1C(C(=O)NC(CC#C)CO)(CC=C)CCC1 49758,Cc1nc(C2CCC2)sc1CC(=O)N(CCCNC(C1(CCF)CC1)=O)CCO 49759,N1(C(CCC(CC)=O)=O)CC2(CCCC2NC(=O)C=CC2CCCN2C)C1 49760,c1(C(N(C2(CC(N3C(C(C)O)CC3)=O)CC2)C)=O)cc(C(N)=O)co1 49761,CC(CCCNC(=O)C(C)c1ccsn1)NC(=O)CN(C)C1CC1 49762,C1(NC(C2(C)C=CCC2)=O)COCCN(C(=O)Cc2ccsc2)C1 49763,N1(C(C=CC)=O)CC(F)(n2cc(COCCO)nn2)C1 49764,n1(CCCC)cc(C(=O)NCCC2(O)CN(C(=O)CC3(C)CCC3)C2)nn1 49765,N1(CC)CCC(C(=O)O)CC12CCC2.N1(C(c2ccccc2)C=O)CCC(C)C1 49766,C1(C(=O)NCC2CN(C(Cc3cc(C)on3)=O)C(C)C2)CCC2(CCOCC2)O1 49767,c1(C(=O)NC2(CNC(C3CC4CCCC4C3)=O)CC2)c(OC(F)F)cccc1Cl 49768,c1(OC)ccc(CC(CC(C)NCC)c2nnnn2C2(C)CC2)c2ccccc12 49769,C=Cc1ccc(C(N2CCN(C(C3C(F)(F)C34CC4)=O)C(CO)C2)=O)cc1 49770,CC1OCCCC1C(N1CCC(CCC(=O)NCCCN2CCOCC2)CC1)=O 49771,C1(C2CC2)(C(N(CC#CC)C)=O)CN(C(C2CCCSC2C)=O)C1 49772,c1(C(=O)NC2(CC=C)CN(C(C3CC=C(C)CC3)=O)C2)ccnc(OC)c1F 49773,n1(CC)ncc(C(=O)N(C)CC2CCN(C(=O)CNC(=O)NC)C2)c1C1CC1 49774,C1(NC(C(C)Oc2ccccn2)=O)(CNC(C2(C(N)=O)CC2)=O)CCOCC1 49775,c1(C(N)=O)cc(=NCCCN(C(=O)CN2CCCCS2(=O)=O)CC2CC2)[nH]cn1 49776,Cc1nn2ccc(C3CC3)nc2c1-c1nc(CC2CC2)nn1C1CC1.C12CC1C2 49777,N1(C(CC2CCC(=O)N2)=O)CCN(CC(=O)NC2CC(OCCO)C2)CC1 49778,n1(C(CC)(C)C)nnnc1C(c1nnc(C(F)(F)F)s1)NCC1COC(=O)N1 49779,c1(C(=O)NC(C)CN(C(=O)Cc2ccc(F)cc2)C)c(F)ccc(Cl)c1F 49780,CC1CN(C(=O)C=C2CCN(C)C2)CCCN1C(=O)CN1CC(=O)N(C)C1=O 49781,c1(OCC(=O)NCC(C)N(C)C(c2ccc(CC#N)cc2)=O)ccc(Cl)cn1 49782,c1(CC(N2C(CNC(=O)C=Cc3ccccc3)CCCC2)=O)cc(F)ccc1O 49783,Cc1cccc2c(C(=O)NCC3CC3NC(=O)CSc3cccc(Cl)c3)n[nH]c12 49784,N1(C(C(N2C(C)CCC2C)C)=O)CCC2(CCCN(C(=O)CCCCF)C2)C1 49785,c1(-c2scc(NC(=O)Nc3ccc(Br)c(OC(F)(F)F)c3)n2)ccc2nncn2c1 49786,N#Cc1cc(CNC(=O)Nc2ccc(C3(C(F)(F)F)CC3)cc2)ccn1 49787,C12(C(N3C4C(NC(c5cc6c(s5)CCC6)=O)C(C4)C3)=O)CCC(O)(CC1)CC2 49788,C1(CNC(CNC(CNC(C2C(C)(C)CCO2)=O)=O)=O)CC2CCCC2C1 49789,N1(C(c2c(C)nccn2)=O)CCC(NC(=O)COC2(C)CCC2)C12CC2 49790,Cc1ncc(NC(c2nnnn2C2COC2)C2(C)CC2(C)C)cn1 49791,CN1CC2(CC2)CC1C(=O)NCCCOCCNC(C1CS(=O)(=O)C1)=O 49792,C1(C(N2CC(C)(CC)OCC2)=O)COC2(C1)CC1(CN(C(=O)OC(C)(C)C)C1)C2 49793,N1(C(C2C(NC(C(C)n3ccnc3)=O)C3CCC2C3)=O)CCc2nc[nH]c2C1 49794,Cc1cccc(CC(=O)NC2CC2CNC(C2CC2CCN(C)C)=O)c1 49795,c1(NC(CSc2ccc(C)cc2)C)ccc2ncc(I)n2c1 49796,c1(C(C)(F)F)csc(C(=O)NC2(CO)CN(C(c3csc(Cl)c3)=O)C2)n1 49797,N(C(=NCC1CC1)NCc1ncc[nH]c1=O)C(C)CCc1ccccc1 49798,c1(C(=O)NC2C(NC(CCOC)=O)CCC2)cc2c(cc1Br)OCO2 49799,c1(C(N(C(CCNC(C2(SC)CC(O)C2)=O)C)C)=O)ccc(C)c(C(C)=O)c1 49800,N1(C(c2n(C)cc(C(N)=O)c2)=O)CC2CC1CN(C(C1(F)CC=CCC1)=O)C2 49801,CC1CC=C(C(=O)NC23CCC(CC2)N(C(=O)CC2CC4CC2C2CC42)C3)CC1 49802,C(=O)(C1=C(c2ccccc2)CCC1)NCC(CC)(C)NC(c1cnnc(C)c1)=O 49803,CC1CCC(CCNC(=O)C(Cc2ccoc2)NC(C2CCC(O)C2)=O)CC1 49804,C(C)(CCC(=O)N(CCCN(C(=O)Cc1cnc(C)o1)C)C)SC 49805,c1(CSC)ccc(SCCCCC(=O)N(C(=O)NC(C)(C)C)C(C)C)cc1C 49806,C(C(C(C)C)NC(c1ccccn1)=O)(C1CCCCC1)NC(CCCC)=O 49807,CN1CC(F)CC1C(N1CCC(C(=O)NCC2CNC(=O)O2)C1)=O 49808,Cc1cnc(NC(=O)C(C2CCCCC2)NC(c2cn(C)nn2)C2CC2)c(C)c1 49809,N1(C(C(C2CCN(C(c3cc(C(C)=O)on3)=O)C2)C)=O)CCc2nnnn2CC1 49810,CCC(CNC(C1(F)C(C)(C)C1(C)C)=O)N=c1[nH]nc(C(F)(F)F)s1 49811,N1(C(C2CCC(C)O2)=O)CCCC2C1CCN2C(c1cccc2c1CC(=O)N2)=O 49812,c1(CC)sc(C(=O)NCC2(C)CCN(C(=O)C(c3cccnc3)C)C2)cc1C 49813,CC1CC2(CC(C(=O)NC3CCN(C(C4CCS(=O)(=O)CC4)=O)CC3F)C2)C1 49814,c1(C(CNCCOc2ccc(C(=O)OCC)cc2)C)cc(F)cc(F)c1 49815,C1(C(=O)NCCOCCC#C)C2CC3C(C2NC(=O)C(C)(C)Cl)C13 49816,C1(C)(CC)CC(C(=O)NC(C)CNC(=O)CC#N)CCO1 49817,c1(C(=O)NC(CCNC(CCc2ncc(C)[nH]2)=O)c2cccs2)ncccc1CO 49818,Cc1nnn(C)c1C(N1CCC(C)(CNC(c2ccccn2)=O)C1)=O 49819,c1(C(=O)NC2CCN(C(C(C)=CC)=O)C2CC)cnn2cccc(Cl)c12 49820,C1(C(N2CC3(CN(C(C4C(c5ccn(C)n5)C4)=O)C3)C2)=O)CCC2(CCOC2)O1 49821,C#CC1CN(C(=O)CN(C)C(C)C)CCN1C(=O)CC1(C2CC2)CC1 49822,N1(c2c(C#N)nccn2)CCCC(C2(NC(C3CCCC(O)C3)=O)CC2)C1 49823,CC1(C(=O)N(CC(O)CO)C2CC2)CCN(C(=O)C(=O)NC2CC2)CC1 49824,CC(O)C(C(=O)N1CCN(C2CCC2)CC1)NC(=O)CC1CC2C=CC1C2 49825,CC(C)(C)C(CNC(C1CC=CC(O)C1)=O)C(=O)N1CC2CCC(CO)(C2)C1 49826,C1(NC(c2cc(C)ns2)=O)CC2C1CCN2C(c1cnn(CCO)c1C)=O 49827,c1(C(N2C(C)(CNC(CC(CC)OC)=O)CCC2)=O)ccc2c(c1)CNC2=O 49828,Cc1cc(C)c(C(N2CC(O)(CCNC(=O)C(C)OCCN(C)C)C2)=O)c(O)c1 49829,N1(C(CC=CC=C)=O)CCN(C(c2cc(C(F)(F)F)ccc2O)=O)C(C2CC2)C1 49830,C1(CCOC)(NC(=O)CSc2nncs2)CCN(C(c2ccc(CO)cn2)=O)C1 49831,CC1CC(CNC(c2ncn(C)n2)=O)CN1C(=O)C(F)=C1CCC1 49832,N1(C(c2c(C)nn(C)c2C)=O)CC(C)OC2(CCN(C(=O)CC3CSC3)CC2)C1 49833,Cc1ccc(C(=O)NCC2(O)CC(NC(C3CCN(C)C3=O)=O)C2)cn1 49834,C1(NC(=O)COC2CC2)CC2CN(C(c3cc(Br)c(F)cc3F)=O)CC2C1 49835,C1(CNC(=O)C(F)C(F)(F)F)CC2CCC(C1)N2C(c1ccc2c[nH]nc2n1)=O 49836,S(=O)(=O)(c1ccc(=NCCOCCCOC)[nH]c1)N(CC(COC)OC)C 49837,C1(CNC(C2CCCCO2)=O)CCCCN1C(C1(CO)CCCC1)=O 49838,N1(C(Cc2cn(CC)nn2)=O)CCCC(CNC(=O)CP(C)(C)=O)CC1 49839,C1(n2cc(-c3c(C)nccn3)nn2)CC2CCC1(NC(=O)Cn1cc(Cl)cn1)C2 49840,N1(C(c2ccc(C(C)=O)o2)=O)CCC=C(C(=O)N(CC(N)=O)C)C1 49841,N1(C(C23CC(n4cc(CCSC)nn4)C2C3)=O)CCN(CCN(C)C)CC1 49842,C1(NC(C#CC2(C)CC2)=O)CN(C(C2CC3(CCC3O)C2)=O)C2(CCC2)C1 49843,C#CCC(C(=O)NC)NC(c1cc(CNC(c2nccnc2C)=O)[nH]n1)=O 49844,C1(O)(CNC(CCOCCN(C)C(c2ncc[nH]2)=O)=O)CCOC1 49845,c1(-n2cc(CN(C(=O)C(O)C(F)(F)F)C(C)C)nn2)cccc(S(C)(=O)=O)c1 49846,C1(C2CC2)(NC(C=CC)=O)CCN(C(C2CCCCN2Cc2ccncc2)=O)C1 49847,c1(OCC)cccc(CN2CCC(CC(=O)NC(c3cnn(CC)c3)C)CC2)c1 49848,CC1(C)CC(F)(F)CCC1C(N1CCOC(CCNC(=O)C2=CCC2)C1)=O 49849,n1(CCC)cc(C(=O)NCC2C(CC)CCN2C(c2occc2C)=O)c(C)n1 49850,c1(OC)ccc(F)c(C(=O)NC2CCCCC2NC(c2cccnc2)=O)c1F 49851,C1(C(=O)Nc2cn(CC(=O)OC)nc2)CCC(NC(=O)CSC)CC1 49852,Cc1cc(C(=O)NC(C)CCNC(=O)CC2OCCCC2(C)C)ccc1O 49853,C1(C(=O)NC2(COC)CN(C(=O)CCc3ccnc(Cl)c3)C2)C2CCC(F)(F)C12 49854,c1(C(N2CC(NC(c3cc(C)ncn3)=O)C(C)C2)=O)csc2c(F)cc(F)cc12 49855,c1(C(=O)NCC(C)NC(C2CCC3(CCC3)CO2)=O)csc(S(C)(=O)=O)c1 49856,CC1(C(=O)NCCNC(=O)CCc2nc(O)n[nH]2)CCc2ccccc21 49857,C1(C(C(N2CC(NC(C(C)c3cccs3)=O)C2)=O)C)CCC(C)(C)CC1 49858,c1(C(N2CCCC(C3N(C(CCCC#C)=O)CCCC3)C2)=O)c(C)nn(C)c1Cl 49859,N1(C(c2cnc(C(=O)OC)o2)C(=O)NCC=C)CCOC(C)(C2CC2)C1 49860,C1(n2cc(CNC(C(C)O)=O)nn2)CCN(C(c2occc2Br)=O)CC1 49861,c1(SC)nc(=NC2CCCN(C(c3ccccc3C(C)(F)F)=O)C2)s[nH]1 49862,C1(CNC(CCC(C2CCC(C)CC2)=O)=O)C(C)CCCN1C(=O)CSC(F)F 49863,c1(C(=O)OC)cnn(CCNCC(CO)NC(=O)CC2(OC)CC2)c1 49864,N1(C(C2(C)N(Cc3c(C)scc3)CC2)=O)C2CCCC1COC2 49865,C=CC1(CC)COCCN1C(c1ncc(Br)cc1Cl)C(=O)NC(C)(C)C 49866,c1(CN2CCC3CN(C(c4c(OC)ccs4)=O)CC3C2)cc2ccccc2nc1C 49867,Cc1ccc(CC(N2CC3(CNC(c4ccc(C)n4C)=O)CCC2C3)=O)cc1F 49868,Cc1cc(-c2cn(C3CCC(=O)C3C)nn2)cc(F)c1 49869,N1(C(C(COC(C)C)(C)C)=O)CCCC(NC(c2cnc(O)c(F)c2)=O)C(F)C1 49870,c1(C(=O)NC(C)CCCCNC(=O)C2CC2)coc2c1COC2 49871,N1(C(CC=CC=C)=O)CC2CC1CC2NC(=O)CCSCc1ccccc1 49872,N1(Cc2c(F)cc(OC)c(I)c2)CCC(C)(C)CC(C)(C)C1 49873,N1(Cc2cc(C)c(Br)cc2C)CCC2CN(c3ncc4[nH]cc(I)c4n3)CC2C1 49874,C1(NC(C2CCC(OC)CC2)=O)CCN(C(=O)C(c2ccnn2C)O)CC1O 49875,N1(C(C2C(=C)C2)=O)CCN(C(c2ncc([N+](=O)[O-])n2C)=O)C2(CCC2)C1 49876,C1(C(=O)NCCc2ncon2)(NC(C2C(CCC)C2)=O)CCSC1 49877,c1(C(=O)NC2C(NC(c3cc(C)nn3C)=O)CC2)c(C)nc(O)nc1C 49878,C1(NC(C(n2cc(Cl)cn2)C)=O)(CO)CCCN(C(C2CC3CC2C2CC32)=O)C1 49879,c1(C(CCOCC)N(C(=O)C(C)O)C)cc(C(F)(F)F)ccc1C(F)(F)F 49880,c1(OC)cc(C=CC(=O)NC23CCCC2CN(C(c2cscn2)=O)C3)ccc1F 49881,c1(C(=O)NC(C)(C)CCCNC(=O)CN2CCCCC2)nccc(Cl)c1Cl 49882,c1(NC(C2CSCCN2Cc2cc(F)c(O)c(Br)c2)=O)ncc(Br)cc1[N+](=O)[O-] 49883,C(=O)(CCCC1CC1)N(C1CCN(C(c2cc(-c3ccccn3)ns2)=O)C1)C 49884,C1(C(N2C(C)(C)CC(NC(c3cc(Cl)ccn3)=O)C2)=O)CN2CCCCC2CO1 49885,c1(C(=O)Nc2c(OC)nsc2)ccc(CNC(C2(C)CCNC2=O)=O)cn1 49886,c1(CC2(C(=O)NCC(C)(C)NC(COCCC(C)C)=O)CC2)cc(Cl)ccc1F 49887,c1(NC(C2C(CNCc3cc(OC)ns3)CCCC2)=O)ccc(O)c(C)c1 49888,C1(CNC(C(CC)(C)OC)=O)C2CCC(C2)N1C(=O)CCc1ccc(Cl)cc1 49889,c1(CC)ccc(C(=O)NCC(C2CC2)N(C(=O)C(N2CCNC2=O)C)C)[nH]1 49890,N1(C(C(CCCC)C)=O)CC2=C(C1)CN(C(C1CCCCC1CC)=O)C2 49891,Cc1cc(Cl)c(C(=O)NC(C2CN(C(c3cnc(S)nc3)=O)CCO2)C)cc1N 49892,N1(C(c2ccc(SC)o2)=O)CCC(NC(=O)Cc2sc(C)nc2C)CC1C1CC1 49893,N1(C(CCC=CC(C)C)=O)CCN(CCNC(C2(C)CC=CCC2)=O)CC1 49894,C1(NC(c2c(C)ncc(C)c2)=O)CCCC12CCN(C(c1cn[nH]c1)=O)C2 49895,c1(CNC(C2CC(C)(C)C2)=O)cccc2c1CCN(C(c1cn[nH]c1)=O)C2 49896,c1(C(C)NC(=O)CN(C(=O)CCC2CC2(F)F)C)nncn1C 49897,C(=O)(C(F)(F)CC)N(CCOCCC(=O)N(C1CN(CCC)C1)C1CC1)C 49898,C1(C(=O)NCC(C(C)C)NC(=O)CCn2cccn2)CCC2(CC2)C1 49899,c1(C(N(C)CC2(CNC(c3cccs3)=O)CC2)=O)nc(O)nc(O)c1N 49900,c1(CN(C(c2cn(-c3scc(CC)n3)nc2)=O)Cc2ccco2)ccc(O)cc1 49901,c1(C(=O)NC2(COC)CCN(C(c3ccccc3)=O)C2)ccc(=O)n(C)n1 49902,N12CCCC1(C)C2=O.c1(CC2CCN(Cc3n(CC)ncc3)C2)ccc(C)cc1 49903,C(CC(F)F)(C(=O)NCC(=O)NC1CCCC1)N(C(c1cncc(CC)c1)=O)C 49904,C(C(=O)N(CCCCCCNC(=O)C=C1CCC(C)C1)C)(C(C)C)OCC 49905,C1(C)(C(N(CCC)CCNC(c2ccc(Cl)o2)=O)=O)SCCCS1 49906,C1(NC(C2CC(CNC(C3C(C)CCOC3)=O)C2)=O)CCCCC1N=[N+]=[N-] 49907,Cc1nn(CC(=O)N(CCC(C(C)C)NC(c2snnc2C)=O)C)c(=O)o1 49908,c1(N2CC(C)NC(=O)C2)nc(N2C3CCC2COC3)nc2c1COC2 49909,c1(N2CCC(NC(c3c(C)cc(OC)cc3C)=O)C2)ncnc2cc(C)[nH]c12 49910,C1(C(C)C)CN(C(c2ccon2)=O)CCN1C(c1nocc1Br)=O 49911,C#Cc1cnc(C(=O)NC(CC2CCC2)C(=O)N(CCC=C)C)c(C)c1 49912,C1(CCC)CN(C(c2cnc(Br)c(OC)c2)=O)CCN1C(=O)CCSC 49913,C(=O)(CC(CC1CC1)NC(C1(CC)CCOC1)=O)NCC(CC)O 49914,N1(C(C2(C)CC2)=O)CC2(C1)CN(C(c1csc(Cl)c1Cl)=O)CC2CO 49915,c1(C(=O)NC(C(=O)NCc2cc(C(N)=O)no2)C2CCCO2)cc(C#N)cn1C 49916,C1(OC)CN(C(c2c(Cl)cccc2Br)=O)CCC1NC(=O)CC1CCCCO1 49917,C1(CNCC(=O)N(CC(C)C)CCC)CCC(n2cc(CSC)nn2)C1 49918,N1(C(COc2c(F)ccc(C)c2)=O)CC2CCN(C(C3CCC(C)O3)=O)CC12 49919,N1(CC(N2CC(O)(CNC(C3(c4cccnc4)CCCC3)=O)C2)=O)CSCC1=O 49920,N1(C(COCC)=O)CC2(CC(NC(=O)CCc3ccc(F)nc3)C2)C1 49921,N1(CC2N(CC)CCC2)CCCC(C(=O)N(C)Cc2nncn2C)CC1 49922,C(C1C(=O)N(CCC2CC2)Cc2ccc(s2)C(=O)N1)OCC.C1CC1 49923,C1(C(=O)NCC2C3CN(C(=O)CCN4CCOC4=O)CC23)CCc2cnnn2C1 49924,c1(NC(C2CC(NC(c3cc4ccccc4o3)=O)C2)=O)cnc2ccnn2c1 49925,CC1CC2(CC(C(=O)NCCC3CCC(NC(=O)CCN4CCCCC4)C3)C2)C1 49926,Cc1cccc(NC(=O)NC2(CO)CN(C(=O)Nc3ncccc3F)C2)c1C 49927,c1(C(N(C(CNC(C(C)OC)=O)C)C)=O)ccc(F)c2c1OCC2 49928,CC(C)C(O)C(C)(C)C(=O)NC1CCN(C(C2CCCC2)=O)CCC1(F)F 49929,Cc1ccc(F)c(CNC2(c3nnnn3CCN3CCOCC3)CC2)c1Br 49930,c1(OC)ccc(C(C)C(=O)NCC(O)CNC(c2cnc(N)c(N)c2)=O)c(C)c1 49931,C(N=c1ccnc(NCC(N2CCCCC2)C)[nH]1)c1c(NC(C)=O)cccc1 49932,C1(NC(C2CC(C(F)F)C2)=O)C2CC3CN(C(c4ccc(F)c(F)c4)=O)C1C3C2 49933,C(=O)(CCCCCC(C)(C)C)N(CCCNC(CCc1ccc(C)s1)=O)C1CC1 49934,c1(OC)ncc(F)cc1C(N1CC2CC(NC(c3ccc(C)s3)=O)C1C2)=O 49935,N1(C(CCCCCC#N)=O)CCCC(C2(NC(=O)C=C3CCC3)CC2)C1 49936,C(CC(C(C)C)NC(C1CCC(=O)C1)=O)NC(C(=O)NCC)=O 49937,c1(C(=O)NC2CN(C(C(CC)N(C)C(C)=O)=O)C2)cccc2cc[nH]c12 49938,C(=O)(C1=CCCCCC1)NC1(CC2CC2)CCN(C(=O)CC2(CO)CC2)C1 49939,C(=O)(CC(CC=C)NC(c1ccnc(O)c1F)=O)NC(C#C)CC1CCC1 49940,C(=O)(C(F)(F)C(O)C1CC1)N1CCC(CN(C)C(C2COC(C)(C)CO2)=O)CC1 49941,c1(OC)cccc(NC(=O)COCCNC(c2csc(C(F)F)c2)=O)c1C 49942,c1(CC(=O)NC(CC)CN(C(C2(C#N)CC2)=O)CC)ccc2scc(C)c2c1 49943,c1(C(=O)NC23CC(C(N4C5(C)CC5CC4)=O)(C2)C3)cc2ccccn2n1 49944,c1(C(=O)NC(COC)CO)cccnc1CNC(=O)COCC(F)F 49945,C1(NC(C(C)(C)C(F)(F)F)=O)CC(C2CCN(C(=O)COc3ccccc3)C2)C1 49946,c1(C(=O)OC)[nH]c(=NCC23CCC(C)(CC2)CO3)sc1Cl 49947,C(C(F)(F)C(F)(F)F)OCCC(N1C(C2(NC(CCC#C)=O)CC2)CCC1)=O 49948,c1(C(=O)NCC(CCNC(=O)CC2CC(=O)NC2=O)O)cnc2[nH]cncc1-2 49949,c1(NCC(CCCC)NC(C2(C)CCCCN2)=O)cnc(C#N)c(C#N)n1 49950,CCCC(CC)C(=O)NC(C)C(CO)NC(c1cc(F)ccc1C1CC1)=O 49951,C1(CNC(C(C)NC(CC)=O)=O)CCN(C(=O)CCCS(N)(=O)=O)CC1C1CC1 49952,c1(OC)ccc(-c2ccnc(C(=O)NNC(=S)Nc3ccc(C)cc3)c2)cc1C 49953,N1(CC)CCCC1CC(=O)NCC#CCNC(=O)CCOCC1CC1 49954,c1(CNC(c2cc(Cl)on2)=O)ccc(C(=O)NCC=CCSCCOC)o1 49955,C1(OC)(OC)C(C(=O)NCC2(C)CCCN2C(C)=O)CC1(F)F 49956,c1(C(=O)NCCCNC(c2cc(C)c(Br)o2)=O)n[nH]c2nccc(Cl)c12 49957,Cc1cncc(C(=O)N(C2CCCN(C(=O)CC=Cc3ccccc3)C2)C)c1Cl 49958,S(=O)(=O)(c1c(Cl)ccc2c1OCCO2)Nc1ncnc2sc(C)c(C)c21 49959,c1(C(N2CC(NC(C34CC(C3)C4)=O)CC(C)C2F)=O)ccc(N)cc1S(N)(=O)=O 49960,Cc1nc2c(C#N)cnn2c(C)c1CCC(=O)NCC1CCC2(C1)OCCO2 49961,C1(NC(C2CCN(CC)C2)=O)CCC12CN(C(=O)Cn1cc(C(F)(F)F)nn1)C2 49962,C1(C(=O)NCCCN(C(c2ccccc2O)=O)CC)CC(=O)N(CC(C)C)C1 49963,C(CC(C)C)(C(=O)NCCOC(C)(C)CNC(=O)Cc1cscn1)NC(C)=O 49964,CCCC(CCC)CC(=O)NC1CC2(C1)CC2Nc1cc(Cl)ncn1 49965,c1(C(=O)NC(CC=C)CNC(=O)Cc2ccsc2C)cc2c(O)ncnc2cn1 49966,c1(CCC)nc(-c2ccc(-n3cncn3)cn2)n(C2CCCSC2)n1 49967,C1(NC(C(CCC)O)=O)CC1C1CCCN(C(c2c(OC)cccc2Cl)=O)C1 49968,c1(N(C)Cc2scc(C(C)C)n2)nc(=NC(C)CC(N)=O)[nH]c2c1CCCCC2 49969,CC1(C)CCN(C(C2C3CCC(F)C23)=O)C1C(=O)Nc1ccc(F)nc1 49970,CCCCC(O)C(=O)NC(CNC(C1CCCSC1)=O)C(C)C 49971,Cc1cc(C(=O)N(C)CCNC(c2cc(Cl)c[nH]2)=O)c2ncccc2c1 49972,C1(NC(C(C(C)O)N(C)C)=O)CCN(C(=O)CC2CC(C(C)(C)C)C2)CC1O 49973,c1(OC)cc(Cl)ccc1CC(=O)N(C(C)CN(C)C(C1CC2CCC1CC2)=O)C 49974,CC1(CNC(=O)C(F)=CC2CC2)CC(NC(c2cn(C3COC3)nn2)=O)C1 49975,c1(OC)c(F)ccc(-c2nc(Cc3ccc(F)c(-c4nc(O)n[nH]4)c3)no2)c1F 49976,c1(N(c2c(N(C)C)cccc2)C(c2cc(C#N)ccn2)=O)cc(Cl)cc(Br)c1F 49977,C(=O)(CS(=O)C(F)(F)F)NC(CC)CNC(=O)Cc1ccno1 49978,CCC(C)(C)CNC(=O)C(C1CCCC1)NC(=O)C=CC(C)(C)SC 49979,c1(C(=O)NCCn2cc(C(=O)NCC(=O)NCC(C)C)nn2)ncccc1F 49980,C(=O)(C(O)CC(C)C)N1C(C=CC(N2CC(O)(CC=C)C2)=O)CCC1 49981,C1(C(N2CC(CNC(c3c(COC)ncs3)=O)(OC)C2)=O)CC12CCOC2 49982,c1(OC)ccc2c(CCC(=O)NC3CC(CNC(=O)CCF)C3)c[nH]c2c1 49983,C(CC(=O)NOCC1CC2C=CC1C2)C1CCN(C(c2[nH]cc(C(N)=O)c2)=O)C1 49984,N1(C(c2nn(CC)c(O)c2)=O)CC2(CCCC2)C1C(=O)NCC1=CCN(C)CC1 49985,C1(OCC)CC(N(C(=O)CN(C)C(C2CC2(C)C)=O)C)C1 49986,N1(C(c2n[nH]c(CC)c2Cl)=O)CCC2(CCC2CNC(=O)C(C)C(C)C)CC1 49987,c1(CCC)sc(C(=O)N(C)CC2(CNC(=O)C(C)(C)O)CC2)cc1CC 49988,C1(NC(c2c(C)noc2)=O)CCCN(C(C2CC(F)(CO)C2)=O)CC1 49989,c1(OCC)cccc(C(=O)NC2C3CC2N(C(=O)CC(C)C2CCCO2)C3)c1 49990,c1(C(=O)NC(C2(O)CCN(C(C(=O)NCC)=O)C2)C)ccc2ncn(C)c2n1 49991,N(C(=NCC1CCCSCC1)NC1CCN(CC(F)(F)F)C1)C(CC)CC 49992,CON=C(C(=O)N1CCCC(CO)(NC(=O)C(C)C2CC2)C1)c1ccco1 49993,C(=O)(CCS(C)=O)N1CC(C(C)NC(=O)CC(c2ccccc2)N(C)C)C1 49994,CCCC(CCCNC(C1(C)CCNC(=O)C1)=O)NC(C1CN(C(C)=O)C1)=O 49995,N1(C(C(c2ccc(CC)s2)=O)=O)CC(NC(C2(C)CCC(F)(F)C2)=O)CC(C)C1 49996,N1(C(C(CCC)CC)=O)CC2(CCCN(C(C3COC(=O)C3)=O)C2)C1 49997,Cc1cccc(Br)c1C(C(=O)NC1CC1)Nc1cnn(C2CCOCC2)c1 49998,c1(C(=O)NC(C)CCCCNC(c2cnc(C#N)s2)=O)cccc2nccnc12 49999,C(=O)(C(C)C(C)S(C)(=O)=O)NCCC(C)NC(=O)C=Cc1ccn(C)c1 50000,CC(C)C(C(=O)N1CCC(C)(C)CC1C(N1CCCC1CF)=O)C(C)C 50001,c1(CN(C)C)ccc(C(=O)NCC2CC(F)CN2C(=O)CSc2cccs2)cn1 50002,c1(C(=O)NCC2N(C(C3CC(=C)C3)=O)CCOC2)c[nH]c2cc(OC)ccc12 50003,C1(N(C(C(CC)n2cccn2)=O)CCF)CCCN(C(=O)C=CC(C)(C)SC)C1 50004,CC1(C(=O)NCC2CC3CCC2N3C(C2(CO)CCC2)=O)CCCNS1(=O)=O 50005,C1(NC(C(C)c2ccsc2)=O)CCN(c2cnc(F)cn2)CC1O 50006,N1(C(c2scc(C)c2)=O)CC2CC2(NC(c2ccnc(C3CC3)n2)=O)C1 50007,C1(C)(CNC(c2c(CC)c[nH]n2)=O)COCCN(C(C2CC2CC)=O)C1 50008,C1(OC)CC(C(N2CC=CC(O)C2)=O)N(C(c2sccc2Cl)=O)C1 50009,Cc1cccnc1CC(=O)NC1CC(C)N(C(=O)CN2CCOCC2)C1 50010,N1(C(C2N(C(C(N)=O)=O)CC2)=O)CCOC2CC12 50011,C1(CC)C(NC(=O)COc2cccc(F)c2)CCN1C(=O)C(C)SC 50012,c1(CC)ncc(C(N2CCN(C(=O)CCn3cccn3)C(CC)C2)=O)c(O)n1 50013,C(=O)(C1=NOC(C)(C)C1)NCC1(F)CN(C(C2CCC(C)O2)=O)C1 50014,c1(OC)nn(C)cc1C(N1CC(C(=O)NC2CCN(CCF)C2)C(C(C)C)C1)=O 50015,c1(C(N(CC(C)NC(C2CCCN2Cc2nnn(C)n2)=O)C)=O)ccc(Cl)cc1 50016,Cc1cc(C(=O)NC2CC(F)(F)CC2NC(=O)C2=CCOCC2)cc(Cl)c1 50017,N1(C(C(C)OCCC=C)=O)CC2CC1(CNC(C1CC(C)=NO1)=O)C2 50018,c1(C(N2CCN(C(=O)OCC)CC2)=O)cc(OC)nc2cc(Br)ccc12 50019,N1(C(C#CC(C)C)=O)CCC2(CCCCC2NC(C2CCc3c[nH]nc3C2)=O)C1 50020,CCC(C)(C(=O)NC1CC1NC(c1nc(=O)n(C)[nH]1)=O)OC 50021,N1(CCC2N(C)CCC2)CC(=O)N(CC2(n3ccnn3)CC2)C1=O 50022,CCCC(C)(CC)C(=O)N1CCC(O)(CNC(c2nnn3c2CSCC3)=O)C1 50023,Fc1cccc(CN=C(NCC(F)F)NCC2CCN2C2CCOCC2)c1F 50024,c1(C(N2CCC3CCN(C(CC(C)(C)O)=O)CC32)=O)c[nH]c2ccccc2c1=O 50025,Cc1ccc(CCC(=O)N(CCCCNC(=O)CC2CCCC(C)C2)C)cc1 50026,c1(COC)nc(=NCC(C2CC2)NC(=O)C(c2cccc(OC)c2)O)s[nH]1 50027,C1(C(=O)NC2(C)CN(C(c3cnn(C(F)(F)F)c3)=O)C2)CC2(CCCC2)CO1 50028,c1(OCC=C)ccc(Cl)nc1C(=O)NC1CCC1NC(=O)C(C)c1ccco1 50029,c1(C(N2CCCC(CN(C(=O)C(O)C3CC3)C)C2)=O)cc(F)ncc1Br 50030,N1(CC(C(N2CC(C)C(CNC(=O)CC(C)(C)C)C2)=O)O)CCSC(C)(C)C1 50031,C1(C(N2CC(CCCC)NCC2)=O)CCOC12CCC2 50032,C(C1CN(C(=O)CC(C)C(=O)OC)CC1C(N1CC(N2CCOCC2)C1)=O)=CC 50033,N1(C(C2N(C(C(C)C)=O)CCCC2)=O)CCC(NC(c2cnc(S)[nH]2)=O)C(F)C1 50034,C(CCN(C)C(c1ccc(CC)s1)=O)(C(C)C)NC(c1cc(CCC)[nH]n1)=O 50035,N1(C(C23CC(C#N)(C2)C3)=O)CCC2(CCN(C(=O)C=Cc3cncs3)CC2)C1 50036,CCCS(=O)(=O)C(C)C(=O)NC1CN(C(c2cc(C)ncc2C)=O)C2(CCC2)C1 50037,CC1CN(C2CCCCC2NCCC2CC2(Cl)Cl)CCO1 50038,C1(NC(=O)Nc2c[nH]nc2C(=O)Nc2ncc(OC)nc2)C2CCCCCC12 50039,C12(NC(C(C3CCCOC3)OC)=O)CC(C(=O)Nc3ccn(C)c3C)(C1)OC2C 50040,Cc1ccc(C(=O)NCC(C)(C2CC2)NC(=O)COCP(C)(C)=O)c(C)c1 50041,c1(-c2ccc(CN(C(c3c(CCC)nccc3)=O)C)cc2)cc(OC)cc(O)c1 50042,c1(NCC(C)(C)N(C)C)cc(Br)ccc1S(=O)(=O)NCC1CCOC(C(C)C)C1 50043,C1(C(=O)Nc2c(NCCC)ccc(Cl)c2)CC2(C)CCCN2S1(=O)=O 50044,C(CCCC(=O)N1CC2CC2(CNC(=O)CNC(c2ccc(Cl)cc2)=O)C1)OC 50045,c1(C(N(C2C(N(C)C(C3CC3F)=O)CCCC2)C)=O)cnc2ccnn2c1 50046,N1(C(CSCCCC)=O)CCC12CN(C(=O)CCC(C)(C)F)C2 50047,C1(C(N(C(C(=O)NCCCOCC=C)C)C2CC2)=O)C(C(C)=O)C1(C)C 50048,C(CCCCC(=O)NC1CCC1O)N(C(=O)Cc1cncnc1)C 50049,N1(C(CN(c2ccncc2)C)=O)CCCCCC1CNC(c1ccccc1F)=O 50050,CC1=C(C(=O)NC2COC3(C2)CN(C(c2scnc2C2CC2)=O)C3)CCS1(=O)=O 50051,c1(NC(CN(C(=O)C(F)OC(F)(F)F)C(CC)C)=O)cc(C)cc2c1NCCC2 50052,CC1CC(NC(c2c[nH]c(C(N)=O)c2)=O)CCN1C(=O)CC1(C)CC1 50053,C(=O)(CCCCCc1cn(CCCF)nn1)NC1C(C)(C)C1 50054,CC(C(=O)N=c1ccn(CCO)[nH]1)C1CCN(C(c2ccc3occc3c2)=O)C1 50055,Cc1nccc(C(=O)NC23CC2CN(C(=O)C#CC2CC2)C3)c1C 50056,CCCCCC(O)C(=O)N1CCCC(CCNC(C2(OC)CCSCC2)=O)C1 50057,C(C(CCOC)NC(=O)CC1CCCC1)NC(COCCC=C)=O 50058,N1(C(N2CCC(N3CCCCC3)C2)=O)CCCC1NC(C1CC(C(F)(F)F)C1)=O 50059,C#Cc1ccc(C(N2CCC(NC(C3(F)CCOC3)=O)C(O)C2)=O)c(F)c1 50060,C#CC1CCC(C(N2CCC(CNC(C3CCC(C4CC4)C3)=O)CC2)=O)CC1 50061,CCCCC(C)CCC(=O)N1CCC(C(=O)NOCCCOCC)C12CC2 50062,c1(C(C)(C)C)cccc(COc2cnc(C3CN(C(=O)OC(C)(C)C)C3)o2)c1 50063,n1(CC)nnc(C(=O)NCCC2(C)CCN(C(C3CCS(=O)(=O)N3)=O)C2)c1C 50064,C1(C(=O)NCc2n(C)ccn2)CC2CCC1N2C(=O)C(C)(O)C1CCC1 50065,n1(CC(=O)N(C2(c3cn(CCOCC)nn3)CCOC2)C2CC2)ncccc1=O 50066,CON1CCC(CC(=O)NC2CCN(C(C3(OC)CCCCCC3)=O)C2C)CC1 50067,C(=O)(C1=C(F)CN(C(C2C3C4CCC(C4)C23)=O)CC1)NCc1ccc(C#N)cc1 50068,Cn1cnc2ncnc(Nc3cc(-c4ccc([N+](=O)[O-])nc4)ccn3)c12 50069,c1(C(=O)NC2CC(NC(C34C(C(=O)OC)(CCC3)C4)=O)C2)ccn2nnnc2c1 50070,c1(C(C(=O)N(C2(C(=O)OCC)CC2)C)NC(N)=O)ccccc1 50071,CC1CCC(CNC(=O)CCC(F)(F)F)CN1C(=O)CC1CCCNC1=O 50072,C1(N(C(C(=O)NCCC#N)C2CC2(Br)Br)C)CC=CCC1 50073,c1(-c2nc(CSC)nn2CC2CC(C)C2)ccc2c(c1)COCC2 50074,Cc1ccc(C(N2CC(F)(F)CC2C(=O)NCCC(C)C)=O)c(O)c1 50075,C1(C(C(c2n(C(CC)(C)C)nnn2)NCCc2ccncc2)C)CC2CCC1O2 50076,N1(CC)CCC1C(=O)NC(C(=O)NCCOCC1CC1)C1CCOC1 50077,N1(C(c2nc(COC)sc2)=O)CC(NC(=O)C2=CCCO2)C(C)(C)C1 50078,CC1(C)CC(NC(c2ccc(Cl)cc2N)=O)CN1C(C1CS(=O)C1)=O 50079,Brc1cc(-c2noc(-c3csc4c3CCNC4)n2)c2c(c1)OCO2 50080,c1(OC)ccc(CC(N2CCNC(C(=O)Nc3c(C)ccnc3Br)C2)=O)cc1Cl 50081,N1(C(C2CC(=O)NC2)=O)CCCC(C2CCN(C(=O)CCc3ccc[nH]3)C2)C1 50082,C1(C(N(CC(CC)(F)F)C)=O)CN(C(=O)CC2CC3(CC3)CO2)CCO1 50083,C1(CNC(CN(C(C)=O)C)=O)CCN(C(=O)CCc2ccncn2)CC1 50084,c1(CC)cn2c(n1)CC(C(=O)N(CCCNC(C1(C(C)C)CC1)=O)C1CC1)CC2 50085,N#Cc1cc(C(N2CCOCC2CNC(c2cnc(C3CCCO3)s2)=O)=O)c[nH]1 50086,N1(C(c2c(CC)occ2)=O)CCCC(C2CN(C(=O)C(C)OCCC(C)C)C2)C1 50087,CCCC(O)CC(=O)N(CCC(C)NC(c1occc1-c1ccc(F)cc1)=O)C 50088,N1(C(C2(CC#C)CCCCO2)=O)CCN(C(=O)Cc2cncn2C)CC(CO)C1 50089,N1(C(CCc2cncc(C)c2)=O)CCN(C(=O)Cc2ccc(C)nc2)CC(O)C1 50090,C1(CNC(C=Cc2ccc(C)o2)=O)CN(C(c2cnn(CCF)c2)=O)CCN1C 50091,N1(Cc2cccc(OC(F)F)n2)CC2CC3CCCN3C2C1 50092,C12(NC(=O)Cc3cc[nH]n3)CCCC1CN(C(c1c(F)cncc1Cl)=O)C2 50093,Cc1cn2ccnc(C(=O)N(C)CC3CCN(C(=O)Cc4cc[nH]n4)CC3)c2n1 50094,c1(C(=O)OCCOC)ccc(CNC(=O)C2CC2)cc1.C12CCCC1(OC)C2 50095,C1(C(=O)NCCN(C(c2ccn(CCF)n2)=O)CC)CC(O)CN1C(C)=O 50096,C1(C)(C(=O)OC)CC(F)(F)CN1C(=O)CC1CNCC(C)(C)O1 50097,C1(C(C)(O)C(N2CCC(NC(C3CCCCC3)=O)CC2)=O)CCC(F)(F)CC1 50098,c1(NC(C2(F)CN(CC3CCCC3)C2)=O)c(Br)cccc1[N+](=O)[O-] 50099,c1(OCOC)ccc(C(=O)NC(C)(C)CNC(C2CCCC23CC3)=O)cc1 50100,Cc1nsc(C(=O)NC(C)CN(C(=O)C(C)Cc2ccccc2)C)c1N 50101,CC(C)(C#N)CCC(=O)N1CCSCC1C(N1CCS(=O)(=O)CC1)=O 50102,c1(CC)cnccc1C(=O)NCC1CCN(C(C2C=CCC2)=O)C1 50103,CC(C(=O)NC1CCCC1NC(=O)C=Cc1c(Cl)cccc1Cl)C(F)(F)C(F)F 50104,C(C(C)(C)SC1CC(OC)C1)(c1nnnn1CCCC(=O)OCC)NCC 50105,C1(NC(c2cccc(SCC)c2)=O)CCN(C(=O)C(C)S(N)(=O)=O)CCC1(F)F 50106,c1(C(=O)NC(C(C)C)CNC(c2ncsc2C2CC2)=O)ccc(Br)cn1 50107,C(C(O)C(=O)NC1(CNC(=O)CC2CC(OC(C)=O)C2)CCOC1)N(C)C1CC1 50108,Cc1nn(CC(=O)N(CC(C)NC(c2n[nH]cc2C(F)(F)F)=O)C)cc1Cl 50109,C12(C(N(C3CCN(C(C(C(C)C)F)=O)C3)C)=O)C3CC(CC13)C2(F)F 50110,c1(CC(N2C(C)(C)CC(CNC(=O)CNS(C)(=O)=O)C2)=O)cnc2n1CCOC2 50111,CC1(C)OCC(CCN=C(NCC2CCCO2)NC2CC=CC2)CO1 50112,C(CS(=O)(=O)NC(=O)CC1CC1C1CCCC1)OC 50113,C(=O)(CCCS(N)(=O)=O)N1CC(N(C(=O)C=CC(c2ccccc2)=O)C)C(O)C1 50114,C1(C(=O)NC2CCCC(NC(c3c(C)cc(F)s3)=O)C2)CC2C(C1)C2(F)F 50115,N1(C(c2c(OC)cccn2)=O)CC2(NC(=O)Cc3ccc(F)cn3)CCC1CC2 50116,CCCC(C)(CCC)C(=O)NC(C)C(C)NC(=O)C=Cc1ccccc1 50117,N1(C(C=C(C)Cl)=O)CC2CCC1(CNC(=O)C(c1ccc(F)c(F)c1)O)CC2 50118,c1(CCC(=O)O)ccccc1Cl.C#CCOCCOCCOCCC1CC1 50119,C1(CN(C(=O)CNC=O)C)CC(F)CN1C(=O)CNC(=O)CCn1ccnc1 50120,c1(OC)noc(C)c1C(=O)NC1COCCC1NC(C1(C2CCCO2)CCC1)=O 50121,CCC(C(=O)NC1CCCC1C(=O)NCC1(CO)CCOC1)SC 50122,C1(C(=O)NCC(C)CNC(C2(C)CCN(C)C2=O)=O)COc2ccc(F)cc2C1 50123,C(C(CC(=O)N1CC2=C(C1)CN(C(C1C3CCC1CC3)=O)C2)C(F)(F)F)N(C)C 50124,S(=O)(=O)(c1cccc(=NCC(O)c2ccccc2F)[nH]1)N1CC(CC)N(C)CC1 50125,C1(CNC(CSCCCC)=O)N(C(=O)C(C)C(=O)OC)CCCC1(C)C 50126,CC(CC(=O)NCC1CC1CNC(c1ccc2c(n1)CCCN2)=O)CC(C)(C)C 50127,CC(C)CCC(C(=O)NCC(CO)C(C)C)NC(=O)CCN(C)CCO 50128,c1(C(=O)NC(CNC(c2c(C)ccnn2)=O)C)cn2cccc(F)c2n1 50129,CCCC(CC)CCC(=O)NC1CN(C(=O)CCc2ccc(N)c(F)c2)CC1F 50130,C(=O)(C(C)(C)Cc1ccccc1)NC(CN(c1nnc(C)s1)C)C 50131,c1(N(C(C2(CNC(=O)OC(C)(C)C)CCCC2)=O)CC)ccc(Br)cn1 50132,C(=O)(C(C)CC(F)F)N.c1(C(N2C(C(C)O)CCC2)=O)cc(OC(F)F)ccn1 50133,C(c1ccc(Br)cc1)=CCOCCOCCNC(C(=O)OC)N(CC(=O)OC)C 50134,C#CCCC(C(=O)NC1CC(O)CC1O)NC(=O)CN1CCC(C)C1 50135,c1(OC)cccnc1C(=O)N(C1CCN(C(C2CCOC2C(C)C)=O)CC1)C 50136,c1(CNC(=O)NCc2n(C)nc(COC(C)(C)C)n2)c(Cl)cnc(F)c1F 50137,C1(C(=O)NCC(C)(C)O)CC2(CC2)CN1C(=O)CN(CCO)CCO 50138,N1(C(CN(C(=O)CC(O)CN(C)C)CCC)=O)CCC(C)(C)C1C 50139,N1(C(C2C(C)C2)=O)CC2(C1)CN(C(C1CCC(=O)N(C)C1)=O)CC2CO 50140,Cc1cnncc1C(=O)NCC(C1CCC1)NC(=O)C(C)Cc1cccc(Cl)c1 50141,C1(OC)CN(C(C)=O)CC1NC(=O)C(C(C)C)n1cnnc1 50142,C(=O)(C(C)C(C)NC(=O)CCN1CCCC1=O)N(C)CC1C(C)OCC1 50143,n1(CC=C)nnnc1C(CC1CC1)(CC)NCc1ccsc1C 50144,c1(C(=O)NCCN2CCN(C(CC(C(=C)C)OCC)=O)CC2)ccc2n[nH]cc2n1 50145,CCC(C)C(CC(=O)N1CCC12CCCSC2)NC(c1cc(F)cc(F)c1)=O 50146,C1(CCNC(C2CN(C(N)=O)C2)=O)CN(C(c2nnsc2C(F)F)=O)CCO1 50147,N1(C(=O)C(c2cccc(Cl)c2)O)CCCC(NC(C2CC(C(F)F)C2)=O)CC1 50148,c1(CC(=O)NCCCN(C(=O)CSc2nc[nH]n2)CCC)cnsc1 50149,CC1CC(NC(=O)C(C)(C)CC2CC2)CN(C(=O)Cc2cncn2C2CC2)C1 50150,C1(NC(C(c2cnn(C)c2)OC)=O)CC12CC(NC(=O)CCCC1CCCC1)C2 50151,CC1=C(C(=O)NC23CCC(C(=O)NC4CC(CN(C)C)C4)(CC2)C3)CCCO1 50152,C=CCC(CNC(C1CCO1)=O)C(=O)N(C)Cc1cccc(F)c1C 50153,Cc1ccc2c(c1)C(C(=O)N1CCCC(CNC(=O)C(C)C)CC1)OCC2 50154,C1(C(=O)Nc2cc(C(=O)OC)no2)COC2(CCN(C(C3CC3(C)C)=O)CC2)C1 50155,C1(N(C(C(CCCC)N(C)C)=O)C)CC2CCC(C1)N2C(c1ocnc1C)=O 50156,c1(C(=O)NCCN(C(=O)CCC2CC2C)C(C)C)cncc(N2CCCC2=O)c1 50157,Cc1c(C(=O)NC(CNC(C2CCS(=O)CC2)=O)C2CCC2)c[nH]c2nccc1-2 50158,N1(C(C=CC2N(C)CCC2)=O)CC(C)(C)CC1C(=O)NC1CCC2(CC2)C1 50159,N1(N(C(c2c(Cl)ncn2C)C)CCN2CCOCC2)CCN(C)C(=O)C1 50160,[N-]=[N+]=NCC(C(=O)NCCN1CCC(CO)C1)NC(c1nnsc1N)=O 50161,C1(NC(C2(CC)CC2)=O)CCC2CCN(C(=O)C(c3ccc(C)cc3)C)C12 50162,C1(NCc2n(C(C)C)cnc2)CCCC(N)CCC1 50163,N1(C(c2c(C)occ2)=O)CC(NC(=O)C(c2cccc(F)c2)O)C(C)C1 50164,c1(OC)cc(C)cc(CN2CC3C(C(=O)NC4CCCCCC4C)C3C2)c1O 50165,C(CCC(C)(F)F)N(C)C(c1sccc1CNC(=O)CC1CCCOCC1)=O 50166,N1(C(C(CC)C2CCC2)=O)CC(N(N(C)S(N)(=O)=O)C(C)(C)C)C2CCCC12 50167,N1(C(CC(C)(C)O)=O)CCC2(CCN(c3ccnc(C4CC4)n3)C2)C1 50168,c1(OC)ccc2[nH]c(CN3CCC(O)CC3C(=O)Nc3csc(C)n3)cc2n1 50169,c1(C(N2C(C)C(NC(=O)CCCC(F)F)CCC2)=O)cnc([N+](=O)[O-])n1C 50170,CC1CN(C(=O)CO)CC(C)N(C(c2cc(Cl)cc(Br)c2F)=O)C1 50171,C=CCC(C)C(=O)N1CCC(CCC(N2CCC(CCC)CC2)=O)C1 50172,C1(C(N2CC(OC)C(NC(=O)CC34COCC(C3)C4)C2)=O)CC2(CCCO2)C1 50173,Cc1cc2ccccc2n1CC(=O)NC1(C)CCN(C(C2(C)CC2C)=O)C1 50174,Nc1cc(C(=O)NCC2CCCN2C(c2cncc([N+](=O)[O-])c2)=O)cc(F)c1O 50175,S(=O)(=O)(c1cccc(=NCc2cnc(N3CCCC3)nc2)[nH]1)NC(C(CC)(C)C)C 50176,N1(C(CSC)=O)CCc2nc(CNC(C3(C)CC3(F)Cl)=O)sc2C1 50177,CC1CCN(C(c2ccc(CNC(=O)C=CC3CC3)nc2)=O)CCS1 50178,c1(OCC)c(C(N2CC(CNC(c3c(C)cccc3Br)=O)C2)=O)cccc1F 50179,S(=O)(=O)(c1ccccc1Cl)NCC(=O)N(C1CC(NC(c2occ(C)c2)=O)C1)C 50180,c1(NC(CCC)CC)[nH]c(=NC2CSCCC2C)nc2c1ncn2C(C)C 50181,N1(C(C(CC)=CC)=O)CCC2(NC(c3nncn3CC)=O)CCCCC12 50182,C1(C(=O)NC(C(=O)NCC(C(C)O)O)(C)C2CCC2)C(C#N)C1(C)C 50183,c1(C(CC)=O)cnn(C)c1Cl.C1(C)(CN)CC(NC(C2(CSC3CC3)CC2)=O)C1 50184,C1(C(=O)NC2CC(C)(NC(C(CC)Sc3ccccc3)=O)C2)CC(F)CN1C 50185,C1(C(=O)NC(C2CCCC2O)C)CCCC1CNC(c1cc[nH]n1)=O 50186,c1(C(N2C(CC(=O)NCc3ccc(F)cc3F)CCC2)=O)ncnc2[nH]cnc12 50187,c1(CC)ccsc1C(=O)N(C)CC1CCN(C(C2CC3CC3C2)=O)C1 50188,Cc1nc2ccnn2cc1C(N1CC(O)(CNC(C2CC2(C)Br)=O)C1)=O 50189,N1(C(C(C)C2CCC2)=O)CCC(CO)(CNC(c2ccnc(Cl)c2N)=O)CC1 50190,C1(C(N(C)CCOCCNC(c2cnn(C3CCC3)c2)=O)=O)CC12CC2(F)F 50191,CCCC(C)C(=O)N1CCC(NC(=O)CC=C(C)C)CC1 50192,N1(C(C(c2cccc(OC)c2)(F)F)=O)CCC2(CC(NC(C3CCCS3)=O)C2)C1 50193,C1(C#N)(CNC(CC2(C)N(C(Cc3nc(C)[nH]n3)=O)CC2)=O)CCCC1 50194,CC1CCCCN1C(C1CC(NC(c2cc(Cl)cs2)=O)C(O)C1)=O 50195,C1(NC(CC2(C)CCN(C(CCC(CC)=O)=O)C2)=O)CCC(=O)N(C)C1=O 50196,c1(C(N(CC(C)(C)NC(=O)C2=NOCC2)C)=O)cc(F)cc2nc(S)[nH]c12 50197,C(C(CC)CCO)NC(CCN(CC#C)C(c1cnc(Cl)s1)=O)=O 50198,N1(C(CCCC#CC)=O)CC2(C1)CN(C(c1cc(C)c(Cl)s1)=O)CC2CO 50199,Cc1cc(C(c2nnnn2C2CC2)NCC(C)(C)C(N)=O)cc(C)n1 50200,C1(c2nnnn2CN2CCOCC2)(NCCc2ncc(C)o2)CC(C)SC(C)C1 50201,C1(NC(c2ccc(C#N)o2)=O)CC(C(=O)NCC2(F)CCC2)C12CCC2 50202,CCCCC(C(=O)NCC(C)N(C)C(c1nc(C(F)(F)F)cs1)=O)C(C)C 50203,N1(C(c2cc(Cl)c3n[nH]cc3c2)=O)CCC2(CCN(C(c3ccco3)=O)CC2)C1 50204,C(=O)(CC1=NNC(=O)C1)NC1CC(OC)CN(C(C(CC)(C)C)=O)C1 50205,CC#CCC(C(=O)NC1CCC12CCCC2)NC(c1ccc(OC)nn1)=O 50206,C(=O)(C(C)C(=O)NCCOCCCNC(C1CNC(=O)C1)=O)OC 50207,C1(NC(C23CCC(OC)C2C3)=O)CN(C(=O)CC2CC3(CCO2)CC3)CCC1O 50208,S(=O)(=O)(c1ccc(C(=O)NCC2CC2NC(c2cnn(C3CCC3)c2)=O)o1)NC 50209,N1(C(C23CC(COC)(OC2)C3)=O)CCCC(N(C)C(C2OCCOC2C)=O)CC1 50210,C1(CC=C)(NC(=O)C2=CCC2)CCN(C(c2ccc(CCC)cc2)=O)CC1 50211,c1(C(=O)OCC)nc(C(=O)NCCN(C(C2COCCO2)=O)CC2CC2)cs1 50212,C(=O)(CCCC(C)(C)NC(c1cnn(CCF)c1)=O)NCC1N(C)CC(O)C1 50213,N1(C(C(COCC)C)=O)CC2CCC(C1)N2C(c1cccc(F)c1O)=O 50214,Cc1nc(C(C)C)sc1C(N1CC(NC(=O)C2=CCC2)CC1CO)=O 50215,c1(C(N(CC(C)N(C(CN(CCC)C)=O)C)C)=O)sc(Cl)c(Cl)c1C 50216,c1(CC(=O)NCCC2(NC(c3cn(C(C)C)nn3)=O)CC2)ccc(F)cc1 50217,C1(C(C)NC(=O)CSCC(N)=O)CCCN1C(=O)CC1(C)CCCO1 50218,N1(C(C2(C(C)(F)F)CCC2)=O)CC(NC(=O)CC2OCCC2(C)C)CC(O)C1 50219,C1(C(=O)N(C)Cc2cncnc2)(CC)CCN(C(=O)C(C)NC(=O)NC)C1 50220,CC1=C(C(=O)N2CCOCC2CC(=O)NC(C2CCC2)C2CC2)CCC1 50221,C1(NC(C=CC(C)C)=O)CN(C(=O)CSC(C)C)CC1C(F)(F)F 50222,C(=O)(C(C)CCCOC)NCC1CN(C(C(c2cccc(Cl)c2)CC)=O)C1 50223,Cc1c(Cl)c(Cn2cc(CCC3CCCCC3)nn2)nc2ccccc12 50224,CCCC(C)CCCC(=O)N1CCCC1C1(O)CN(C(c2ccc(C)nc2)=O)C1 50225,c1(NC)c(C(N2CCC(N(C)C(c3csc(CO)n3)=O)C2)=O)cccc1F 50226,c1(OC)cccc(CNC2CC2C(=O)Nc2cc(C(C)(C)C)on2)c1C 50227,c1(C(=O)NCC2CC(C)N(C(c3cscc3C(F)(F)F)=O)C2)ccnc(C#N)c1 50228,CCCC(C(=O)NC1COCCN(C(=O)C(CC)CC)C1)C(C)C 50229,N1(C(C2CCC(C)(C)O2)=O)CCC2CN(C(=O)CCCC#N)CC2CC1 50230,N1(C(C2=CN=C2C(F)F)=O)CCN(C(c2cc(C3CC3)sn2)=O)C(C2CC2)C1 50231,C(=O)(C1(Nc2c(Br)cccc2S(C)(=O)=O)CCc2c(OC)cccc21)OC 50232,C(CCC(C)C(C(=O)Nc1ccc(Cl)cc1F)N(C)CC1CC1)=C(C)C 50233,CC(CNC(c1nnn(CCO)c1N)=O)CC(F)F 50234,c1(NC(C(C)CSC(F)(F)F)=O)cccc(-c2cn(CCCN(C)C)nn2)c1 50235,c1(C(=O)OCC)ccc(CC(N2CCC2C(=O)Nc2cc[nH]c(=N)c2)=O)cc1 50236,N(C(=NCCN1CC2CCC1C2)NC1CCS(=O)(=O)C1)Cc1scc(C#N)n1 50237,O=C(C1=CCC(NC(c2n[nH]c(O)n2)=O)C1)NC(CC1CC1)C1CC1 50238,CCCC(F)(F)C(=O)NCC1CC1CNC(=O)CCn1cncn1 50239,C(=O)(C(C)(C)C(=O)NC1CC(NC(=O)C(C(C)C)n2cc(Br)cn2)C1)OC 50240,N1(CCC(C)C2CCCO2)CC(=O)N(Cc2c(I)cnn2C)C1=O 50241,C12(NC(CCCOC(C)=O)=O)CCC(CC1)N(C(C)=O)C2 50242,c1(C(N(C2CCCN(C(=O)CCc3cocn3)C2)CC)=O)cc(F)cnc1O 50243,C1(CNC(CCC(C)OC)=O)(NC(C2CCC(F)(F)C2)=O)Cc2ccccc2C1 50244,c1(SCC(=O)NCCN(C2CCCC2)C(C=CC(CC)=CC)=O)n[nH]c(C)n1 50245,C12(NC(c3cc(CCC)[nH]n3)=O)CCC(CC1NC(=O)C(C)n1cncn1)C2 50246,c1(SCC(=O)NCC(CNC(CCOCCCC)=O)C)nnnn1C1CC1 50247,Cn1cc(C(N2CC(NC(C34CCOC3CCOC4)=O)C2)=O)c2cccnc12 50248,C1(NC(C2CC2C(F)(F)F)=O)CCC2CCN(C(c3coc4ccccc34)=O)C12 50249,CC(Cc1cccs1)CN=c1[nH]c(=NCCN2CCCC2C)[nH]c2c1CSC2 50250,c1(C(=O)NC2CCN(C(=O)CCOC3CC3)CC2)c(F)ccc(F)c1F 50251,C(CCCCC(=O)NCC1CCN1C(=O)CCn1cnc([N+](=O)[O-])c1)NC(N)=O 50252,CC1CN(C(c2cnc(O)cc2O)=O)CC(CCNC(c2ccn(C)c2)=O)O1 50253,c1(C(N2CCC(COC)(NC(=O)C(O)C3CC3)CC2)=O)cc2cccnn2c1 50254,CC(C(=O)N1CCC(CO)(CNC(=O)C(C)NC(N)=O)C1)S(N)(=O)=O 50255,CC#CCCCC(=O)NNC(=O)Nc1ccc(C(N2CCOCC2)C)cc1 50256,N1(C(C(=Cc2cn[nH]c2)C)=O)CCN(C(c2csc(C(F)(F)F)n2)=O)CCC1C 50257,N1(C(C(=CC2CCCC2)C)=O)CC2OCCN(C(=O)CCS(C)=O)C2C1 50258,CCCCC(C(=O)NC1CCCCCC1C)NC(=O)C=CCN1CCCC1 50259,C(=O)(CCC(C)S(C)(=O)=O)NCC1CC(NC(CC(C)C(F)(F)F)=O)C1 50260,Cc1cc(CC(=O)NC2CC(C)(CNC(c3c(C)cccc3F)=O)C2)cc(F)c1 50261,Cc1ncc(C(N2CC(O)(CNC(=O)CC3CCC3(F)F)C2)=O)c(=N)[nH]1 50262,c1(CCC)ccccc1C(=O)NC(C1CN(C(c2cc(CC(C)C)on2)=O)C1)C 50263,C(=O)(CCCCNC(C)=O)N1CC(C(=O)NCC2(OC)CN(C)C2)(OC)C1 50264,Cc1ccc2[nH]c(C(N3CC4CCC4(NC(C4(F)CCOC4)=O)C3)=O)cc2c1C 50265,N1(CCCN(C)C2CC2)CC2(C(=O)NC3CCCCCC3)CCCC2(F)C1 50266,C(CC(O)CNC(c1cnn(C2CC2)c1)=O)NC(C(N1CCCC1=O)C)=O 50267,C1(CN(C(Cc2cc(C)ns2)=O)C)CCCN(C(c2occc2Cl)=O)C1 50268,C=Cn1nncc1C(=O)Nc1cccc(NC(=O)CC(O)c2ccccc2)c1 50269,C(C(N=[N+]=[N-])C(=O)N1CC(=O)CC1C(=O)NC1(CC(N)=O)CC1)OCC 50270,N1(C(c2nc(N(C(C)=O)C)sc2)C2CC2)CCC(=O)N(Cc2cccnc2Cl)C1=O 50271,N1(C(C2CCC([SH](CC)CC)C2)=O)CCN(CCN(C)C(C2CCN2CC)=O)CC1 50272,C1(CC)(NC(=O)CC2CCC(=O)O2)CCN(C(=O)CCCn2ccnn2)CC1 50273,C1(S(C)(=O)=O)(C(=O)NCC2C(CNC(CSC)=O)C2)CCCCC1 50274,c1(OC(CC)C)ccc(C(=O)NCC2C3CN(C(C4CC=CCO4)=O)CC23)cc1 50275,C=CC1(CC(=O)NCC(C)N(C)C(C2CC(=O)NC(C)C2)=O)CCCCC1 50276,Cc1cccc2c(C(N3CCCN(C(=O)CSC(C)C)C(C(C)C)C3)=O)n[nH]c12 50277,N1(c2ccc(CC)cc2)Cc2ccc(NC(=O)NC(CNC)C(C)(C)C)cc2C1=O 50278,N1(C(C2(C#C)CC2)=O)CCC2(CCCCN(C(C3CCC4(CCC4)CC3)=O)C2)C1 50279,Cn1nc(C(N2CC3CC3(CNC(c3ccncc3N(C)C)=O)C2)=O)cc1O 50280,C(=O)(C1c2c[nH]nc2CCC1C)N1CC2N(Cc3cc(C)on3)C(CC2)C1 50281,C(=O)(CCC(C)(C)NC(=O)CC1(C)CCCC1)NCC(C)NC(=O)OC 50282,c1(C(N2CC3C(NC(C(CCC)OC)=O)(C3)C2)=O)ccc(Br)cc1F 50283,C1(N(C(CCC(=C)Cl)=O)C)CN(C(=O)C(CC(=C)C)NC(C)=O)CC1(C)C 50284,S(=O)(=O)(c1cc(C(=O)NC(C)CCN(C(=O)C=C2CCCCC2)C)c(C)o1)NC 50285,C(=O)(CS(=O)(=O)N1CCN(CCCNC(C2(C)CC2F)=O)CC1)OCC 50286,N1(C(c2ccnc(C)n2)=O)CCC(C)CC1CNC(=O)COCCCC(C)C 50287,C1(C)(CNC(C)=O)CCN(c2nnnn2CC(C2COC(C)(C)O2)(C)C)CC1 50288,CN1CC(C(N2CC(O)(C(F)C(=O)NCC3CC(O)C(O)C3)C2)=O)CCC1=O 50289,c1(C(=O)NCC(CC)NC(C(CCC)O)=O)cccc(S(=O)(=O)NCC(N)=O)c1 50290,c1(CCCn2cc(-c3c(C)noc3C)nn2)c(C)nn(C)c1C 50291,C(=O)(CC(O)CC(C)(C)C)N(C(CC(C)C)C(=O)NCC1(F)CCN(C)C1)C 50292,c1(CC(N2C(C)CC(CNC(=O)CC3CC(N(C)C)C3)C2)=O)ccc(F)c(F)c1 50293,c1(CC(N2CC(NC(C3C(CC)C3)=O)C(C)C2)=O)cc(SC2CC2)cc(F)c1 50294,N1(C(C(C)O)=O)CCN(C(c2cc(C3CCCN3C)[nH]n2)=O)CC1 50295,c1(OC)cccc(C(=O)N(C)CC2CN(C(c3cnco3)=O)CCO2)c1OC 50296,CS(=O)(=O)c1ccccc1CN1CC2C(C1C(N1CCCC1CO)=O)C2(C)C 50297,C(=O)(C1CCc2cc(Cl)ccc21)N1CC(NC(c2nc(C)n(C)c2)=O)C(F)C1 50298,c1(C(=O)NCC(CC=C)NC(=O)COC(C)CC)cc2nc(OC)ccc2[nH]1 50299,C1(NC(C2N(C(C)=O)CCC2)=O)CC(NCC2CCC3(CC2)CC3)C12CCC2 50300,c1(C(N2CCC(NC(c3n(CC=C)ccn3)=O)C2C)=O)ccc2c(n1)CCCC2 50301,c1(CC)cc[nH]c1C(=O)NC1CCC1C(=O)NCCn1cnc(CO)c1 50302,c1(CNC(Cn2c(C)ccn2)=O)cccc(NC(C2CCCCC2C)=O)c1 50303,c1(C(=O)NC2CCN(C(COCC)=O)C2(C)C)cc2c(Br)c(C)ccc2[nH]1 50304,C1(N(C)C)CN(C(C2CSCCS2)=O)CC1CNC(c1csc(CO)n1)=O 50305,N1(C(C(C)C)=O)CCC(C)CC1CNC(c1ccc(SCCCO)cc1)=O 50306,C1(C(=O)OCc2c(C)occ2)CN(C(=O)OC(C)(C)C)C(C)CO1 50307,C1(C(N2CC3CC3(C(N3CCC(n4cncn4)C3)=O)C2)=O)CC2CC1CC2O 50308,c1(CC)ccc(Br)cc1C(=O)NC1CC(N(C(=O)CC2CCOCC2)C)C1 50309,c1(C(N2CC3CC2CN3C(C2CC3(CCCO3)C2)=O)=O)ccc(Cl)cc1Cl 50310,C1(NC(CCN(C)CC)=O)CCCN(C(c2cc(C)n(C=O)n2)=O)C1C.C1CC1 50311,CCCCC(C)(F)C(=O)NCC1CC(NC(=O)CC2(N(C)C)CCCC2)CCO1 50312,Cc1onc(Cl)c1C(N1CC2C(CNC(c3snc(Cl)c3Cl)=O)C2C1)=O 50313,N1(C(C)C)CC(NC(=O)CN2CCN(C(=O)Cn3ncccc3=O)CC2)CC1=O 50314,C1(NC(C=C(C)C(C)C)=O)C2CC1N(C(=O)Cn1cc(C)cn1)C2 50315,C(CC(CC)C(=O)NCCOC1CCN(C(=O)C(C)NC(N)=O)CC1)=CC 50316,c1(C(N2CCCC(CCNC(C(COCC)(C)C)=O)C2)=O)cnc2scc(C)n12 50317,N(S(=O)(=O)N1CCC2(CCCCC2)CC1)CC(CCCC)OC 50318,C1(C2CCN(C(=O)CC3=CCCC3)CC2)(NC(CC2(N(C)C)CCCC2)=O)CC1 50319,N1(C(C(C)N(C)C)=O)CCC(N(C)C(c2ncc(C(F)F)s2)=O)CC1 50320,N1(C(C(C)OC)=O)CC2(CC(NC(c3cn4cc(C)ccc4n3)=O)CO2)C1 50321,C1(C(=O)NCC2N(C(c3n[nH]c(CC)c3Cl)=O)CC(O)C2)CCOC(C)(C)C1 50322,c1(COC)nc(C)c(C(=O)NCCCC2CCCN2C(=O)CN2CCC2)s1 50323,N1(C(C2(c3cn(C)nc3)CCCO2)=O)CC2CS(=O)(=O)CC2(C(=O)O)C1 50324,C1(CC(=O)Nc2ccccc2)(N(C(=O)CSC(F)(F)F)CC2CC2)CCOC1 50325,C1(CNC(CCC2C(C)(C)C2)=O)(NC(c2ccc(=N)[nH]n2)=O)CCCCC1 50326,C1(C(=O)NCC(C(C)(C)C)NC(c2c(CC)c[nH]c2)=O)CCCCC(=O)N1 50327,c1(OC)cc(OC)c(OC)cc1COC.c1(-n2ncc(CN(C)C)c2)ccc(C)cc1 50328,CCCCC(C)(C)NC(C1(NC(=O)CN2CC(C)(C)C2)CC(F)(F)C1)=O 50329,N1(c2c(Cl)cnc(OC)n2)CCC(C2(NC(=O)CCSC(F)(F)F)CC2)CC1 50330,c1(OC)ccc2c(c1)C(C(=O)Nc1ccc(C(=O)NCCC(C)(C)O)cc1)CC2 50331,n1(CC)cc(C(=O)NC(C)CC(C)NC(=O)CN2CCNC(=O)C2)c(C(C)C)n1 50332,C1(OC)CCCC(C(=O)NCCCN(C2CCCC2)C(c2cn(C)c(C)n2)=O)C1 50333,C(N=c1[nH]cnc(Cl)c1F)C1C(NC(CCCn2c(C)ncc2)=O)CCCC1 50334,CCC(CC)CCC(=O)NCCC1(C)CCN(C(C2CC(OC)C(OC)C2)=O)C1 50335,C(=O)(C(F)C(=O)NC(C)(CSC)C(=O)NCC=C(C)C)OCC 50336,C(=O)(C(C)(CCC)CCC)NCCC(=C)CNC(=O)COC(C)=O 50337,N1(C(CC#N)=O)CCC2(CC2C(=O)Nc2cc(C(F)F)no2)C1 50338,c1(C(N(C(CNC(C=COCC)=O)C)CC)=O)ccnc2ncnn12 50339,c1(OC)ncc(C(=O)NC(C)(C)CN(C)C(C2CC3(CSC3)C2)=O)cc1Cl 50340,C(c1cc2ccccc2n1C)=CC(=O)NC(C)CNC(c1cc(Cl)ns1)=O 50341,C(=O)(CCCC(C)(C)C#N)NCC(CNC(CSCC)=O)F 50342,N1(C(CCCC#C)=O)CC2CCCC1C2CNC(=O)CC=C 50343,c1(COC)ncc(CNC(N2CCCC(c3n[nH]c(=N)o3)C2)=O)c(=N)[nH]1 50344,c1(C(=O)NCC(C2CC2)NC(c2nncn2C2CC2)=O)ccncc1C(F)F 50345,N1(C(c2cc(C#C)c(Cl)cc2)=O)CCC2(C1)CN(C(=O)CCN(C)CC)CCO2 50346,N1(C(C(C)=C2CCC2)=O)CC(C(N2CCC(C(C)(C)C)C2)=O)(SC)C1 50347,Cc1cnc(NCc2cscc2C)c(S(=O)(=O)NC2CC3CC(CO)CC23)c1 50348,c1(C(N(CCN(C(=O)CC(C)(C)CC)CC)CC)=O)cc([N+](=O)[O-])c(C)cc1C 50349,c1(C(=O)NC2CC(CNC(C(C(C)c3ccccc3)O)=O)C2)ccnc(F)c1O 50350,C1(C)(C(=O)NCCC(C)N2CCCC2)CCCN(C(C2CCOC2(C)C)=O)C1 50351,CC(C)C(O)C(C)(C)C(=O)NC1COCC1C(N1CC(C)(CF)C1)=O 50352,c1(CNC(c2nnnn2CCC2CC2)(CC)C2CCC2)cccc(C(C)(F)F)c1 50353,C1(NC(CCC)=O)CC(CNC(=O)CCCOC(C)C)C1(C)C 50354,N1(C(C23CCC(NC(CCCCSC)=O)(CC2)C3)=O)C2CCC1CC(CO)C2 50355,N1(C(CCOC)=O)CCC(C(F)(F)F)CC1CNC(c1cnn(CC(C)C)c1)=O 50356,C1(C(=O)NC(C(C)C)CCN(C)C(C2CC2(F)F)=O)CC1C1CCCCC1 50357,CCC(C)CCC(=O)NC1(c2cn(C(c3cccc(F)c3)C)nn2)CC(F)(F)C1 50358,Cc1ccc(C(O)C(N2CCCC(NC(c3ccc(Cl)nc3)=O)C2)=O)cc1 50359,CC(CN(C)C)CC(=O)NCC1C2CC1N(C(C1COCCN1C)=O)C2 50360,N1(C(C(CC)(C)COC)=O)CCCCC(CNC(=O)Cc2ccc(C)cc2)CC1 50361,c1(CNC(C2CC2NC(c2[nH]cc(CC)c2)=O)=O)cc(OC)c(OC)c(OC)c1 50362,C1(CC#C)(C(=O)NCC(O)C(F)F)CCN(C(=O)CCCC#N)C1 50363,c1(C(C(=O)NCCCOC)N(CCC(N)=O)CC2CC2)nc(C#N)cs1 50364,Cc1cc(C(=O)NC2(CC(=O)Nc3nnc(C)o3)CCC2)nc(C)c1 50365,Cc1cnc2c(C3C(NCCC(=O)O)CC3OC(C)(C)C)nccc2c1 50366,C(C)(C)(CC(F)C(=O)NC1(c2ncc(C)o2)CC1)NC(c1c(CC)nn(C)c1)=O 50367,c1(C(N2C(CN(C(c3nccc(C)n3)=O)C)COCC2)=O)cc2c(ncn2C)[nH]1 50368,c1(C(=O)NC2C3CN(C(c4ccn(C(C)(C)C)n4)=O)C2C3)n[nH]c2c1COCC2 50369,C1(NC(c2sc(C)c(O)n2)=O)CC2CC(C1)N(C(C1(C)CCCCC1)=O)C2 50370,c1(C(C)C)nc(C(=O)NCC2C(NC(=O)Cc3cnns3)CC2O)co1 50371,c1(-n2cc(CN3CCCC(NC(c4ccno4)=O)C3)nn2)ccc2c(c1)CCO2 50372,C(=O)(C(C)(F)F)NCC(C)CN(C)C(c1ccc(CSC(F)F)o1)=O 50373,CC1CN(C(C2CC2c2cn[nH]c2)=O)CCCN1C(c1csc(C(F)(F)F)c1)=O 50374,CC(CCCNC(c1nc(Cl)cs1)=O)NC(=O)C(C)(C)c1cscn1 50375,C1(COC)(NC(=O)CC2CCCC2C)CN(C(=O)CSc2n[nH]c(C)n2)C1 50376,C(C)(CSc1ccn(C)c1C)(C(C)C)NC(=O)NC1N(C(CCCC)=O)CSC1 50377,c1(OC)ccc(N)c(C(N2CCOCC2CNC(=O)Cc2cc(Cl)cs2)=O)c1 50378,C1(C(N2CCN(CC(=O)NC(c3cscn3)CO)CC2)=O)CC12CCCCC2 50379,CC1N(C(C2N(C(c3ccc[n+]([O-])c3)=O)CCC2(C)C)=O)CCOC1(C)C 50380,c1(C(N2CCC(N(C(C(CC(C)C)C)=O)CCO)C2)=O)nn2cccnc2c1Cl 50381,Cc1cnc(CC(=O)N(C)CC2CCCN2C(=O)C(C)CC2CCC2)o1 50382,c1(C(N2CCCCC3CCC23)C(=O)NCCOC)ccc(F)c2ncccc12 50383,C1(CC)CNC(=O)CN1C(=O)CC1CN(C(=O)Cc2cccc(C)c2)CC1C 50384,CC1(C)CN(C(c2ccc[nH]2)=O)CC1C(=O)NCc1ncco1 50385,Cc1ccc(Cl)cc1C(N1CC(NC(c2ccc(Cl)nc2O)=O)CCC1C)=O 50386,C(=O)(C1=C(C)OCCS1)NCc1nc(CNC(CC(CCC)C)=O)sc1 50387,CN1CCC(CC(=O)NCCC2CCN(C(=O)C(C#N)=CC3CC3)CC2)C1=O 50388,C1(C)(CNC(CN2CCC(C)CC2)=O)COCCN(C(c2cnsn2)=O)C1 50389,C(=O)(CCC(=O)NCC(CC)NC(C1CCCN1c1ncccn1)=O)NCC 50390,C(=O)(C1=COc2ccccc2O1)CCNC.C12(C(=O)NCCO)CCCCC1C2 50391,c1(SCC2(C3CN(C(C(C4CCCC4)OC)=O)C3)CC2)ncccn1 50392,CC1CN(c2cccc(Cl)c2)CCN1CCCc1cccnc1 50393,N1(C(c2cn(C)cn2)C(=O)NCC(C)C)CC(C(N)=O)C2(CC2)C1 50394,C#CC1(C(=O)NC2CC3CCCCN3C2)CCN(C(c2c[nH]c(C#N)c2)=O)CC1 50395,c1(CCC(=O)NC(CC2CN(C(C(CC)(C)F)=O)C2)C)c(C)nn(C)c1C 50396,C1(CC(=O)NCC(CNC(=O)Cn2cc(C3CC3)cn2)OC)CCC(=O)NC1=O 50397,Cc1cc(I)c(Cl)cc1N(C(=O)C(C1CCCNC1)O)Cc1ccncc1 50398,C(=O)(C(C)(C)C(=O)N1CCOCC(C(N2CCN(C)C(CO)C2)=O)C1)N(C)C 50399,N1(C(COC(C)C)=O)CCN(C(=O)Cc2cncnc2)C(CS(C)(=O)=O)C1 50400,CCCC(CNC(c1cc(C(F)F)[nH]n1)=O)C(=O)NCCC1(C)CCCO1 50401,C(CCCC(=O)NC1CCC(NC(C2(C)CSC2)=O)C1)SC 50402,C(=O)(CC(C(F)(F)F)OCC)N1CCC(CC=C)(NC(=O)COCCCOC)C1 50403,N1(C(CC(C)CNC(=O)CCc2ccc[nH]2)=O)CC2(CNC(=O)N2)C1 50404,C1(NC(C(C)C(=O)OC(C)(C)C)=O)CN(C(=O)CCCCc2cnc[nH]2)CC1(C)C 50405,CC1Cc2cc(OCc3ccc(C(C)C(F)(F)F)cc3)ccc2O1 50406,CN1C(=O)CSC1=CC(=O)NCC1CC2CCC1N2C(=O)CN1CCCCC1=O 50407,Cc1ncc(C=CC(N2CCC3CN(C(c4cc(C)nn4C)=O)CC23)=O)c(O)n1 50408,N1(C(CCc2cc(OC)no2)=O)C2CCC1CC(NC(C1CC(=O)N(C)C1)=O)C2 50409,Cc1ccc(C(=O)NCC(=O)NCCC(O)CNC(C23CC(CO2)C3)=O)s1 50410,c1(CC(=O)NCC(C)N(C(=O)Cc2nccn2C)CC)ncc(F)cn1 50411,C1(C(=O)NC2(CNC(C3(F)CCS(=O)(=O)C3)=O)CC2)CC(c2ccccn2)=NO1 50412,C1(CC(=O)OCC)CCN(C(c2cccc(Br)c2Cl)C(=O)NCCSC)C1(C)C 50413,c1(NC(C(=O)Nc2c(C(=O)NCCC)cccc2)=O)ccc2c(c1)SCC2 50414,N1(C(C(C=CC)O)=O)CCN(C(=O)CSCCCc2ccccc2)C2CC12 50415,CC1CC(CNC(=O)C#CC(=O)NC2CC2)CN1C(C1CC(=C2CCC2)C1)=O 50416,N1(C(c2c(OCC)cccc2Cl)=O)CCC2(CC(NC(=O)CC(F)(F)F)CO2)C1 50417,c1(OC)ccc2c(CC(=O)NCC3CCN(C(C4(C)CCC4)=O)C3)coc2c1C 50418,c1(CC)ccc2c(c1)OCC2C(=O)N1CCC(C)C(F)(F)CC1 50419,C(=O)(CCC[N+](=O)[O-])NC(C(C)C)CCNC(=O)CCn1ccc(=N)[nH]1 50420,c1(C(=O)NC(CNC(CNS(CC)(=O)=O)=O)(C)C2CCC2)cccc(F)c1Cl 50421,CC1(NCC(CC2CC2)CO)CS(=O)(=O)C1 50422,CS(=O)(=O)C1CCC(CNC(=O)C(=O)NC2CCC(F)(F)CC2)CC1 50423,C(CC(C)C)(C(=O)NC(C1CCCCC1)CNC(=O)CN1CCN(C)CC1)OC 50424,CC(C)CC(C)(O)C(=O)N1CCN(C)C(C(=O)NCCCc2cncnc2)C1 50425,c1(C(N2CCC(N(C(C(CCOC)C)=O)CCO)CC2)=O)c[nH]c2nccc-2c1 50426,CCC(CC(=O)N1CCN(C(=O)C(=Cc2cccnc2)C)C2(CC2)C1)C(F)F 50427,c1(C(=O)NCC2C=CC(NC(C=CCCC)=O)C2)c(OCC)cc(OC)cc1N 50428,c1(C(=O)NCC2CCS(=O)(=O)C2)cc(-c2cccnc2C2CC2)cc2c[nH]nc12 50429,C(=O)(CC1OCCc2ccsc21)NCC1C(C)CCCN1C(=O)Cc1cccs1 50430,CC1CCN(CC(N2CC(CNc3ccnc(-c4ccccc4Cl)c3)C2)=O)CC1 50431,N1(C(C=C(C)C(C)(C)C)=O)CCOC(CCNC(=O)CN2CC(C)C2)C1 50432,Cc1cc(CCC(=O)NCC2CC(NC(=O)Cn3nccn3)C(O)C2)nn1C 50433,c1(C(=O)NCC2(NC(C(Br)=C(C)C)=O)CCC2)cn(C2CC2)nn1 50434,C12(NC(C=C(C)C3CCCCC3)=O)CCCCCC1N(C(C1COC1)=O)CC2 50435,c1(C(=O)NC(C)CCNC(=O)CSc2nnc(S)s2)cc2cccnc2[nH]1 50436,Cc1nc(O)sc1C(=O)NC1CCOCC1C(=O)NCCC1CC(F)(F)C1 50437,Cn1c(COC(C2OCC2(C)C)=O)ccc1Cl 50438,c1(C(=O)NC2CN(C(C3(C=C)CC3)=O)CC2C)ccc(NC(=O)OC)cc1Cl 50439,c1(CC)ncc(C(N2CCC(CF)(NC(=O)CC3C=NN(C)C3=O)C2)=O)c(O)n1 50440,C1(CNC(C(CC#C)C2CC2)=O)CN(C(c2cccn2CCC)=O)CC12CCC2 50441,CCC(C(=O)NC(C)(C)C=CC(=O)NCC1CCSC1)n1ccnc1 50442,c1(-n2c(-c3c(CC)cno3)nc(C3CCC3)n2)ccc(C)cc1OC 50443,CCC(C)CC(=O)C(=O)N(C(C)C(=O)NCCc1cc(C)on1)C1CC1 50444,C1(CC(N2CC(C)(C(=O)NCC3(F)CCOCC3)C2)=O)(OC)CCOCC1 50445,C1(NC(C2CC(=C)C2)=O)CC(CNC(c2ccc(NC3CC3)nc2)=O)C1(C)C 50446,c1(C(=O)NC(CNC(CN(C)CC)=O)C(C)C)cn2c(n1)SCC2 50447,S(=O)(=O)(c1nc(N2CCC(C(C)(C)CO)CC2)ccc1Br)NC(CC)CO 50448,c1(C(=O)NCC2(C)CCN(C(C3CCCCO3)=O)C2)ccc2cnsc2c1 50449,N1(C(C2C(=C)C2)=O)CCCCCC1CNC(c1cc(C(C)C)nn1C)=O 50450,C1(CC(=O)N(c2cc(CCOCCO)on2)CCSc2cccs2)CCCCO1 50451,c1(CC(=O)N(CC(CC)OC)C)ccccc1CNC(=O)CN1CCCNC1=O 50452,c1(C(=O)NCc2c(C(=O)Nc3ccc(CCC)cc3)c[nH]n2)cc2occc2[nH]1 50453,c1(N(C)C)ccccc1N(C(=O)C(=O)NCC(=O)Cc1ccccc1)C 50454,C(=O)(C(C)C(O)CCCC)NC1(CC(=O)N(CCCCCC=C)C)CCCCC1 50455,Cc1ccc2nn[nH]c2c1NC(=O)N=c1cc(C2CCCO2)[nH][nH]1 50456,Cc1c(C(=O)N(CC(O)CNC(=O)CCc2nncn2C)C)nn(C)c1Br 50457,C1(CC(=O)NC2CC(c3n(C)ccn3)OCC2)CC2(CCOCC2)CCO1 50458,N1(C(=O)Cc2ccccc2F)CCC(CCCNC(C23CCC2C3)=O)CC1 50459,N1(C(CC(C)F)=O)CCN(C(c2csc(CO)n2)=O)CC1c1ccc(F)cc1 50460,N1(C(C(CCCC=C)NC(=O)CCC(C)(C)F)=O)CC(C)OC2(CCC2)C1 50461,C1(C(=O)NCC2N(C)CCC2)CCCC(NC(C2(CO)CCCC2)=O)CC1 50462,N1(C(C2C(C(=O)OC)CCCC2)=O)CC(NC(=O)CCCN2CCC2)CC(C)C1 50463,C1(C(N2C(C(N(CCn3c(C)ncc3)C)=O)C(C)C2)=O)CCCC(C)(C)C1 50464,C12(C(=O)NCC#CCNC(c3cc(C)nc(O)n3)=O)OCCCC1C2(F)F 50465,C1(COC)CCCCN1C(c1ccc(C)s1)C(=O)Nc1ccc(C)nc1 50466,c1(C(N2CCC(NC(c3c(C(C)C)[nH]cc3)=O)C(C)C2)=O)cccc2cnnn12 50467,c1(C(N2CCC(NC(C3CC34CCC4)=O)(CF)C2)=O)cc2c(Br)cccn2n1 50468,N1(C(=O)C2=CS(=O)CCC2)CCOCC2(COCCN2c2nc(Cl)ncc2F)C1 50469,CCS(=O)(=O)CC(=O)N1CCN(C(=O)CN2CCSCC2)CC1C 50470,c1(NC(c2c(C(C)C)scn2)=O)cc2c(cc1Br)CCC(=O)N2 50471,N1(C(C2C(CC)C2)=O)CCC(O)(CN(C)C(c2ccc(CC3CC3)cc2)=O)C1 50472,CC1CN(C(=O)CC2C(C)(C)C2(C)C)CC1NC(c1ccc(C2CC2)o1)=O 50473,c1(CC)cnccc1C(N1CCOC(CNC(c2c[nH]c(=NC)s2)=O)C1)=O 50474,N1(CC(CC(C)C)N(CC(F)(F)F)C)CCNCC(O)C1 50475,c1(C(=O)NCC2CC(OC)CN2C(c2cncc(Br)c2)=O)cn2c(n1)CCC2 50476,CC1(C)CCCCC1(C)NC(c1cccc(CNC(c2cscn2)=O)n1)=O 50477,N1(C(C(CC)O)=O)CC2CCC(NC(c3ccc(C(F)(F)F)cc3)=O)C2C1 50478,c1(C(=O)NCCCN(C(CC2CC(OC)C2)=O)C(C)C)cnn2ccc(C)nc12 50479,CCN(Cc1ccn(C)n1)N1CCCC1c1ccc(Cl)c(Cl)c1 50480,c1(C(=O)NCC=C2CCN(C(CC(C)C3CC3)=O)CC2)cc(Cl)cc([N+](=O)[O-])c1 50481,C1(NC(=O)CCCC2CCCC2)CC2(C1)CC2C(=O)NOC1CCOC1 50482,c1(C(=O)NCCCCCCO)cc2cc(-c3cnc4nccn4c3)ccn2n1 50483,N1(C(CCCCC#C)=O)CCC2(CC1)CC2CNC(c1c[nH]ccc1=O)=O 50484,C1(N(CCC2CC2)CC)CCCN(Cc2ccc(F)cc2)C1=O 50485,N1(Cc2cccc(OC)c2)C(=O)CN(CCc2ccnn2C)C1=O 50486,CC1CN(C(=O)CCP(C)(C)=O)CC1(C)C(N1CCCC(CN=[N+]=[N-])C1)=O 50487,c12ccoc1CNC2C.c1(CNC(C2(CCC)CCC2)=O)noc(C(C)(C)C)n1 50488,C(C)(CN=c1[nH]c2ccccc2cc1C#N)N(C(C=C1CCC(C)CC1)=O)CC 50489,c1(NC(C2CCN(C(=O)CCC3CCC3)CC2O)=O)cncc(Cl)c1Br 50490,C(=O)(C1=NOC2(CCC2)C1)NCC(CN(C(=O)CCSc1cccs1)C)(C)C 50491,c1(C(C)(C)C)cccnc1C(N1CCC(CNN(C2CC2)C2CC2)CC1)=O 50492,C1(NC(C(CC2CCC2)OC)=O)CC2CCC1N2C(C1CNC(=O)O1)=O 50493,N1(C(CCCCOC)=O)CCC(C2CCN(C(=O)Cc3c[nH]ccc3=O)C2)CC1 50494,c1(C(=O)NC23CC(NC(C45CCCC4CC5)=O)(C2)C3)cc2ncccc2s1 50495,Cc1ccncc1C(=O)N(C)CCOCCN(C(=O)Cc1cscc1F)C 50496,CCC(CC)C(F)C(=O)NCCN(C(=O)Cn1cnnn1)C 50497,Cc1ccc([N+](=O)[O-])c(N2CC3CCCN(C(c4oncc4C)=O)C3C2)c1 50498,N1(C(C2(COC)CC=CC2)=O)CC2CC(NC(=O)CCOC3CCOCC3)C1C2 50499,c1(C(=O)NC2C(C)CN(C(=O)C=CC(C)(C)C)C2)nn(C)cc1S(C)(=O)=O 50500,N#CC1(CC(=O)NC2CCOC(CNC(=O)C=CC3CC3)C2)CCCCC1 50501,c1(Cc2nnn(CC(F)(F)F)n2)nc(O)c2cnn(C)c2n1.CN1CCN1C 50502,c1(CN2C3CN(C(c4ccc(N(C)C)cc4)=O)C(C3)C2)ccc2cc[nH]c2n1 50503,C1(C(=O)NCC(C)NC(=O)CCCC(N)=O)CC12CCC1(CC2)OCCO1 50504,c1(C(N(C2C3CN(C(c4cnc(C5CC5)[nH]4)=O)CC23)C)=O)ccc(O)nc1Cl 50505,C1(C(C)(C)NC(C2CN(C(C)C)C2)=O)CCN(C(=O)Cc2nncn2C)CC1 50506,c1(CNC(N2C(CC)C(=O)NCC2)=O)ccc2c(c1)cc(C)n2C 50507,C(C1CN(C(=O)CC2CCN(C)C2=O)CC1C(=O)NCC(F)C1CCC1)=CC 50508,c1(NC(C2N(C(C3(COC)CCC3)=O)CCC2)=O)nnc2ccc(Cl)nn12 50509,O=C(NN1CC(C(F)(F)F)C1)C1CC=CCC1NC(=O)Cc1cn[nH]c1 50510,CCC(C)C(CC(=O)NOCC(O)C(C)C)NC(c1cccn1C1CC1)=O 50511,c1(-c2ccc(NC(Cc3ccc(OC)cc3)=O)cc2F)cc(F)cc(F)c1O 50512,C(=O)(CCCC(=O)N1CC2(CNC(=O)CC3(C)CC(F)(F)C3)CC1CO2)N(C)C 50513,c1(N(C(C)C)C)ncnc2sc(Br)cc12.c12ccc(cc1)N(C)C2 50514,c1(C(N(CC(CNC(CSCC(C)C)=O)C)C)=O)cc([N+](=O)[O-])c[nH]1 50515,c1(C(=O)NC2CCN(C(C3=C(CC)OCCS3)=O)C2)cccc2nc(O)n(C)c12 50516,c1(NC(C2CCCN(C(=O)CSc3cccc[n+]3[O-])C2)C)ncc(C#N)cc1Cl 50517,N1(C(COCC#C)=O)CC2CC2(C(=O)NC(COC(C)C)CC)C1 50518,Cc1cnc(C(=O)NCC2CN(C(C34CC(F)(CO3)C4)=O)C2)cc1Br 50519,C1(NC(C2(C)CN(C(=O)CC3CC4CCC3C4)C2)=O)CCC(C2CC2)C1 50520,C1(O)(C(=O)NCCN(CCOC)C(c2c(C)cccc2C)=O)CCCC(C)(C)C1 50521,C1(NC(C(C=C)(C)C)=O)CCCC2CN(C(c3cnc(SC)nc3O)=O)CC12 50522,C1(C(=O)NC2(CO)CN(C(C(C)(C)C3CCCC3)=O)C2)CCCCC1F 50523,N1(C(C(F)OC)=O)CCC(CCN(C)C(c2cnn(C(C)C)c2N)=O)CC1 50524,C1(CC#C)(C(=O)NCC2CCN(C(=O)C(c3ccccc3)C)C2)CCCC1 50525,n1(CC(=O)NC2(C3N(C(CC(C)F)=O)CCC3)CC2)cc2ncccc2n1 50526,N1(C(c2ccc(=NC)[nH]c2)=O)CCCC2(NC(c3nc(F)ccc3Cl)=O)CC2C1 50527,C#CC(CC(C)C)NC(=O)C(C)CN(C(=O)C(C)(C)CC)C 50528,CN1CCCC12CN(C(C1(C(=O)O)CCN(C(=O)OC(C)(C)C)CC1)=O)C2 50529,c1(OC)ccc(C(N2CCN(C(C3CCC(C)CC3)=O)CC2C)=O)c(OC)c1C 50530,C(CC(C(C)C)NC(c1cccc(-n2cncn2)n1)=O)N(C(C(C=CC)O)=O)C 50531,C(CN=c1nc(OCC)cc(C)[nH]1)NCCOCC.C1(C(=O)OCC)CCCCC1 50532,C(CCSC)(C(=O)NCCC1(OCC)CCC1)NC(CCC#C)=O 50533,c1(CC)cccc(C(N2CCC(N(C)C)(CC)CC2)C(=O)NC2CCOC2)c1F 50534,c1(C(N2CC3CC3(C(=O)NCCc3cc[nH]n3)C2)=O)c(F)ccc(F)c1Cl 50535,N1(C(Cn2ccc(C)n2)=O)CC2(CC2)CC1C(=O)NCC1CCCO1 50536,c1(C(=O)NC(CC2CN(C(C3CC(CCC)C3)=O)C2)C)cc(C)nn1C 50537,C12(NC(C3(S(C)(=O)=O)CC3)=O)CCOC(CNC(C3CC3C3CC3)=O)(C1)C2 50538,c1(C(=O)NCC2(O)CN(C(C(C)NC(=O)NC)=O)C2)ccc2cc[nH]c2c1 50539,Cc1cccc(C(=O)NC2CCCCC2CC(=O)NC(c2cccnc2)C)c1N 50540,C1(CC(=O)NCc2ncccc2F)COCCN(C(c2n[nH]c3c2COC3)=O)C1 50541,c1(CNC(=O)NC2(C)C(C)OCC2)ccc(S(N)(=O)=O)cc1 50542,c1(C(N2CC(F)CC(NC(c3ccc(C)s3)=O)C2)=O)cc(O)c(O)c(Cl)c1 50543,c1(C(=O)NC(C2CN(C(=O)C=CCN(C)C)C2)C)ccnn1C1CC1 50544,C1(CC)CCCCC1C(=O)NC1CCCC1CN(C)C(C1CC(F)(F)CS1)=O 50545,n1(CC)cc(C(=O)N(C2CCN(C(=O)C(O)COCc3ccccc3)C2)C)nn1 50546,N1(C(c2cnc(C)[nH]2)=O)CC(NC(=O)CCNS(=O)(=O)c2cccs2)CC(C)C1 50547,N1(C(Cc2cnc(C)s2)=O)CCCCC(NC(c2cnnc(Cl)c2)=O)C1 50548,N1(C(Cc2c(C)cco2)=O)C2CCC1CN(C(C1CCC(C)(F)CC1)=O)C2 50549,N1(C(c2cc(C)nnc2)=O)CC(=O)NCC1C(=O)NC(CN(C)C)C(C)C 50550,C1(C(=O)NCCCCC2CN(C(C3CCC(C(=O)OC)C3)=O)C2)CC12CCOC2 50551,N(C(=NCCc1ccccn1)N1CCCC(O)CC1)CC(C(=O)OC)C 50552,C(C(C)C(C)C(=O)N1CC(C(C)NC(c2ccc(F)cc2F)=O)C1)OC 50553,CCC(C)CCC(=O)NCC12CC1CN(C(=O)C=CSCc1ccco1)C2 50554,N1(C(c2c(C(C)(C)C)ncnc2)=O)CC2(C1)CN(C(=O)CC1CCC(C#N)C1)C2 50555,N1(C(C=C2CCN(Cc3c(C)nc(F)cc3)CC2)=O)CCN2CCOCC2C1 50556,C1(CC(N2CCC(COC)(NC(=O)CCCF)C2)=O)CN2CCN1CC2 50557,N1(C(c2c(OC)ccs2)=O)CCN(C(c2cnccc2Cl)=O)CC1C 50558,C1(CNC(CC2ON=C(C)C2)=O)(CNC(c2cncc(Cl)c2)=O)CC12CCC2 50559,c1(C(N2CC(COC)(NC(=O)CN(C(=O)C(C)C)C)C2)=O)ccc2c(n1)CCOC2 50560,C1(NC(C(C)(C)C2CCOCC2)=O)CC(F)CN(C(C2C3COCC23)=O)C1 50561,Cc1c[nH]cc1C(N1CCC(NC(c2ccsc2-n2cnnn2)=O)C1)=O 50562,Cc1cnn2ccc(C(=O)NC3(C4CCCN4C(=O)C(O)CC(N)=O)CC3)nc12 50563,N1(C(C2=C(C)CCC2)=O)CC2CCCC(CNC(c3cc(C)cs3)=O)C2C1 50564,C(N(O)C(=O)C(O)Cc1cc(F)c(Cl)cc1Cl)c1cn(-c2c(OC)cccc2)nn1 50565,C=C(C)CCC(=O)NC1CCC(CCNC(c2nccnc2C)=O)C1 50566,N1(C(=O)Cc2cc(Cl)ccc2O)CC2CCC1C(CNC(C1(CCO)CC1)=O)C2 50567,n1(CC(N2C(C(CNC(C)=O)Cc3ccccc3)CCC2)=O)cc(F)ccc1=O 50568,c1(C(CN(c2ccc(CC(=O)OC)cc2)C(C)C)=O)c(N)cc(F)cc1Cl 50569,C=C(Cl)C(C)(C)C(=O)N1CC2(CC)CC1(CNC(=O)C(C)NC(=O)C(C)(C)C)C2 50570,c1(C(N2CCCCC(NC(C(COC)OC)=O)CC2)=O)nc2n(c1Cl)CCCC2 50571,O=C1CC2(C1)CC1(CC(NC(C3CCC(c4ccccc4)C3)=O)C1)C2 50572,N1(C(C=CC)=O)CC2CCCC1C2CNC(=O)CNC(C1CCC1)=O 50573,Cc1occc1CC(=O)NC1CC1CNC(c1nocc1-c1ccccc1)=O 50574,C1(CC)CCCN(C(c2cc(CNC(=O)C(c3ccn(C)n3)C)nn2C)=O)CC1 50575,c1(C(=O)NC(C2CCCCC2)C(N2CC(O)C(O)C2)=O)ccn2nccc2c1 50576,C(=O)(C(C)(CO)NC(=O)C(C1CCN(C(=O)CC2CCOCC2)C1)C)OC 50577,N1(C(c2ccc(SCC)nc2)=O)CC2CC(C1)C2NC(=O)Cc1ccccc1F 50578,N1(C(CC2(COC)CCCCO2)=O)CCC2(CCC(NC(=O)C3CC3)C2)CC1 50579,N1(C(Cc2ccc(C#C)cc2)=O)CC2CCC(C1)N2C(C1CC1C(=O)OC)=O 50580,c1(C(N(C)Cc2ccccc2)=O)ccc(S(=O)(=O)NCC2CC2C#N)o1 50581,N1(C(c2c(OC)cccc2O)=O)CCOCC(NC(c2n[nH]cc2I)=O)C1 50582,c1(C(N(C(CNC(C2(NC(C)=O)CC2)=O)C2CC2)C)=O)cc2c(nn1)CCC2 50583,C1(C(=O)NC(COC(C)=O)CO)N(C(=O)CCOCC=CC)CCCC1(C)C 50584,c1(C(N(CCN(C(=O)C(O)C(F)F)C(C)C)C)=O)cc(Cl)ccc1C(F)(F)F 50585,Cc1ccc(C(N2CC(c3ccccc3)(NC(c3cnc(S)[nH]3)=O)C2)=O)cc1 50586,N1(C(C(C(C)O)(F)F)=O)CCC2(CC1)CCN(C(C1(CCN(C)C)CC1)=O)CC2 50587,C1(CNC(C2(C)CC3CC3C2)=O)CCN(C(=O)C(O)C2CCC2)CC1(F)F 50588,c1(N(C)C)ccc([N+](=O)[O-])c(C(=O)NC2CN(C(C3CCC3(F)F)=O)CC2O)c1 50589,C1(C(=O)NCC(C#C)OCC)(CO)C=CCN1C(=O)CCOCCOC 50590,CC1(C)CC(CNc2cc(N3CCOC(c4ccc(F)cc4)C3)ncn2)CO1 50591,c1(C(CNC(C(=O)Nc2cn(CC#C)nc2)=O)(F)F)ccc(Br)cc1Cl 50592,C1(CNC(c2c(CC)noc2C)=O)CCN(C(c2c[nH]c(C)c2)=O)CCC1(F)F 50593,N1(C(CC(C)F)=O)CCCC(CNC(C2(F)CCCCC2)=O)CC1 50594,CC(CF)CC(=O)N(C(C)CNC(=O)C(c1ccc(Cl)cc1)(F)F)C 50595,c1(C(=O)NCC(C)NC(c2c(F)ncc(OC)c2)=O)ccc(F)c(C)c1N 50596,C1(COCC)CCCN(C(CC2CCC3CC23)C(=O)NC2CC2)C1 50597,CCC(C)(C(=O)NC1CN(C(c2ccccc2C)=O)C(CC)(CC)C1)OC 50598,c1(C(N2CCCC2N2CCC(O)C2)C(=O)NCC2CC2)cccc(C2CCC2)c1 50599,c1(CC(=O)NCCc2c(C)ocn2)ccnc(Cl)c1F 50600,C(=O)(C(CC(C)C)NC(C)=O)N(C1C2CN(C(C3(CO)CCCO3)=O)CC12)CC 50601,c1(C(=O)NC(CN(C(c2c(COC)nn(C)c2)=O)C)C)cc2cc(Cl)ccc2s1 50602,c1(C(=O)NC2(CN(C(C3CC(C)NC(=O)C3)=O)C)CC2)ccc(Cl)c(F)c1N 50603,c1(CC)ccc(C=CC(=O)NC2CN(C(=O)CCN3CCCC3)CC2SC)o1 50604,CC(CS(C)(=O)=O)C(=O)N1CCN(C(c2cc3c(ccn3C)s2)=O)C(COC)C1 50605,C1(OC)CC(NCC(=O)OCCOc2ccc(C)cn2)C12CCOCC2 50606,c1(CCC(N2CC(NC(CSCCCC)=O)C2)=O)cc2ccccc2o1 50607,C1(C(=O)NCC(CCC)C)(C(C)C)CCN(C(=O)C(CO)NC(N)=O)C1 50608,Cc1cc(C)n(CC(N2CC(N(C(=O)Cc3c(C)noc3Cl)C)C2)=O)c(=O)n1 50609,c1(C(=O)NCC2CC(F)(CNC(c3cncs3)=O)C2)cc2cccnn2n1 50610,C1(CNC(C(CCC)NC(N)=O)=O)CCCN(C(=O)C2=NNC(=O)C2)CC1 50611,c1(OC)ccc2c(CC(C)NC(c3cnn(CCF)c3)=O)c[nH]c2c1 50612,c1(CN2CCN(C3CCN(C(=O)CC4CCCC4)CC3)CC2)cccc(F)c1Br 50613,C1(C(N(C)CC2(C)CC2)=O)CC(C)(NC(=O)Cn2cc(CO)nn2)C1 50614,c1(COC)ocnc1C(c1nnnn1CC1CC1)NC(CF)CF 50615,c1(CC(=O)NCC(CNC(c2c(CC)nco2)=O)OC)ccc(CO)c(C)c1 50616,C1(NC(c2cnc(C3CC3)[nH]2)=O)CC2CC1N(C(c1csc(Cl)c1Cl)=O)C2 50617,c1(C(N2CC=CC(O)C2C(=O)O)=O)cnc2[nH]ccc2n1 50618,N1(C(Cc2cc(C)ncc2)=O)CCC(C)N(C(c2cccc3nsnc23)=O)CC1 50619,N1(C(c2n(C)c(=O)ccc2)=O)C2CCCC1CN(C(C1CCC13CCC3)=O)CC2 50620,Cc1cccc(C)c1CS(=O)(=O)NC(C1CCC(F)(F)C1)C 50621,C1(CC)(CC)CC(NC(c2cnn(C)c2SC)=O)CN1C(=O)CC1CCOC1 50622,C1(NC(Cc2c(C)ocn2)=O)CN(C(C2CN(C3CCCCC3)C2)=O)CC12CC2 50623,Cc1nc(-c2c[nH]c(C(N3CCC3CNC(=O)CC3CC4(CC4)C3)=O)c2)cs1 50624,N1(C(C(CN(C)C)(C)C)=O)CCC2(CCN(C(=O)CC3CCCCC34CC4)C2)C1 50625,C1(CC(=O)N(CC(=O)NCCOC(CC)CC)C2CC2)CC2C=CC1C2 50626,n1(CC(=O)NC2C(NC(C3(C)C(C)C3)=O)CCOC2)ccc(=O)n(C)c1=O 50627,CC1CCC(C2CCCC2)CN1Cc1cn(CC(C2CCCNC2)O)nn1 50628,c1(OC)ccc(Cl)cc1C(N1CCC(NC(=O)CC2(C(F)(F)F)CC2)C(O)C1)=O 50629,N1(C(CC2(C=C)CCC2)=O)CC2CC2(CNC(=O)CC2CCC(=O)N2C)C1 50630,c1(C(N(C2CCN(C(=O)C=Cc3cn[nH]c3)CC2)C)=O)cc(O)cc(C#N)c1 50631,COn1cnc(C)c1C(N1CC(C)(NC(c2ncncc2C(=O)OC)C)C1)=O 50632,C(=O)(CC(C)CC(C)C)N1C(CNC(c2cccc(C(=O)OCC)c2)=O)CCC1 50633,C(=O)(C1CCc2c[nH]nc21)N1C(CNC(Cn2c(C)ncc2)=O)C(C)(C)CCC1 50634,N1(C(CSC)=O)CC2CCC2(CC(=O)Nc2csnc2C)C1 50635,C(=O)(C1CCCc2scnc21)N(C1CN(C(COCCOCC)=O)C1)C 50636,Cn1nc(C(=O)NC2CCN(c3nc(C4CC4)ns3)CC2O)c2c1CCCC2 50637,C1(CNC(COC(C)=O)=O)C(C)CCCN1C(C1CCCC(F)C1)=O 50638,C1(CNC(CCC2N(C)CCCC2)=O)CCN(C(c2ccc[nH]2)=O)CC1O 50639,CC1(NC(=O)C(O)C(C)(C)C)CCN(C(=O)Cn2cnnc2)CC1 50640,C(=O)(C(C(C)O)NC(=O)CC1CCCN(C)C1)N(C1CC(C)C1)C 50641,C1(C(N(CCCNC(=O)COC2CCOC2)C2CC2)=O)CC=CCC1 50642,Cc1noc2nc(C(=O)NC3CCCN(C(=O)CC4CNC(=O)C4)C3)ccc12 50643,CC(c1ccccc1)=CC(=O)NC1CC1NC(=O)C(C)n1cccn1 50644,C1(NC(=O)CSC2CC2)CC2CN(C(c3cccc(-n4cccc4)c3)=O)CC12 50645,C1(COC)CN(C(C2(C)CCCCO2)=O)CCN1C(=O)CN1CCC(O)CC1 50646,N1(C(C2(C)CNC(=O)C2)=O)CC(C(N2CC3C=CC3C2)=O)C(F)(F)C1 50647,c1(C(N2CCC(Nc3ccc(C#N)cc3)CC2)=O)cc(Cl)sc1S(N)(=O)=O 50648,c1(CN2CCC(C)(CNc3ncn(C)c3C(F)(F)F)CC2)ccc(C#N)c(F)c1 50649,c1(N(CCOC)C)nnc(CN(S(C)(=O)=O)C)n1CC(C)C 50650,c1(N2CCN(C)C(CNC(c3cn4c(n3)CCC4)=O)C2)ncnc2[nH]ccc12 50651,c1(C(C(=O)N(CC(C)(F)F)C)NC(C(C2CCC2)OCC)=O)ccccc1 50652,C1(C)(C(=O)OC)CNCCN1Cc1ccncc1 50653,c1(NC(C(c2ccc(Cl)o2)N(C2CCC2)C)=O)ccc(Nc2ccccc2)cc1 50654,CN(CCNS(C)(=O)=O)N1CC(CO)OC2(CCC2)C1 50655,n1(CC2CC(C)C2)nc(COc2cnn(C)c2)nc1-c1cc(C2CC2)[nH]n1 50656,C1(NC(C=C(C)Cl)=O)CCCCC12CCN(C(=O)C=Cc1ccoc1)CC2 50657,N1(C(CC2C(C)(C)C(NC(=O)CNC=O)C2)=O)CC(O)C2(CCCC2)C1 50658,c1(CC)cc(C(N2CCCC2CCC(C)C)C(=O)NCCC#N)ccc1Cl 50659,Cc1nc2ccc(C(N3CC4C(N(C)C(C56CCCC5C6)=O)C4C3)=O)cc2[nH]1 50660,C12(CNC(c3ccn(CC(F)F)n3)=O)CC1CN(C(C1CC=CC1)=O)C2 50661,CCC(O)C(C)(C)C(=O)NCC(=O)NC1C2CCCC1CCC2 50662,c1(OC(C(=O)NCCC(C)N(C(c2n(CC)ncc2)=O)C)C)cccc(CO)c1 50663,c1(C(=O)NCC2CC(C)N(C(=O)CC3CCCO3)CC2)ccc2c(n1)CCC2 50664,CCN(NC(=O)C(O)CCn1cc(CO)nn1)C(=O)OC(C)(C)C 50665,C1(C(N2CC(c3onc(C)n3)C2)=O)CCOCC1NC(C12CC(C#N)(C1)C2)=O 50666,N1(c2nnc(-c3c(Br)c(C)n(C)n3)n2C)CC2CS(=O)(=O)CC(C1)O2 50667,CCCC(CC)CC(=O)N1CCCCC(NC(c2cc(C3(Cl)CC3)n(C)n2)=O)C1 50668,C1(NC(C(C)CC(N)=O)=O)CC12CCN(C(C1(O)CCCCCC1)=O)CC2 50669,C1(COC)CN(C(C2(CC(F)(F)F)CC2)=O)CCN1C(=O)CCS(C)=O 50670,N1(C(=O)NC(C)CCc2ccccc2)CCN(S(=O)(=O)N2CCOCC2)CC1 50671,CC(C)(C)S(=O)(=O)CC(=O)NCC1CCN1C(C1(C)CCC(=O)N1)=O 50672,C1(C(=O)NC2(c3onc(C)n3)CC2)CCCCCCN1C(=O)C(C)CC#N 50673,CCCC(CCNC(=O)CCC1(C)CN(C(C2CCC(O)CN2C)=O)C1)CCC 50674,C12(C(=O)NCC(C(=O)NCCCN3CCCC3C)OC)C(=O)C3CC1C2C3 50675,c1(OC)c(CNC(=O)C(C2(O)CN(C(=O)C=Cc3cnn(C)c3)C2)F)cnn1C 50676,C(c1ccccc1)=CCCN1CC(CNC(C2N(C(C)=O)CCC2)=O)C1 50677,C1(CNC(Cc2ccc(C)s2)=O)CCC2(CN(C(c3ccccc3O)=O)C2)O1 50678,CCC(CC(=O)N(C(c1ccc(F)c(-c2ccncc2F)n1)=O)CC)C(F)F 50679,N1(C(C2C(C=C)C2)=O)CC(O)(CNC(=O)CC2COCC2O)C1 50680,Nc1cnc(C(=O)NC2COCC2NC(=O)CC=Cc2ccccc2)c(Cl)c1 50681,C=CC(C)(O)C(=O)N(C1CC1)CC1CCCN1C(=O)CC(CC)OC 50682,CC#CCC(C(=O)NCCC(O)CCC)NC(=O)COc1ccccc1 50683,c1(OC(C(=O)NC(C(C)NC(C23CSC(C2)C3)=O)(C)C)C)ccccc1Br 50684,N1(C(CCCOCC=C)=O)CCN(C(CNC(c2cc(C)cs2)=O)C(F)F)CC1 50685,C(=O)(CC(CC)C(C)(C)C)NC(C(=O)Nc1cnc(CCC)nc1)CC=CC 50686,c1(C(N2CCC(NC(CC(CCC)C)=O)C2)=O)cc2c(nc1O)CCC(F)(F)C2 50687,n1(C(CC)C)cc(-c2nc(C(C)Oc3ccccc3)no2)c2ccccc12 50688,Cc1c(NC(=O)C(c2ccc(O)nc2)N2CCCC2C2CCOC2)cccc1Cl 50689,N1(CC=CC(=O)NC(C)C(C)NC(C2CN(C3COC3)C2)=O)CCOCC1 50690,C(=O)(C(F)C(F)(F)F)NC1CC1.C12(CC=CC1)C(=O)NCCC(C)N(C)C2 50691,C=CCCCCCC(=O)N1CC2CC(NC(c3cc(C)oc3CC)=O)CC2C1 50692,C=CCCCCC(=O)NC(C1CCN(C(=O)C=C(Cl)Cl)C1)C 50693,c1(C(=O)NC2(CC=C)CN(C(=O)CS(=O)CC)C2)cnc(F)c(C)c1 50694,C1(C(CNC(C2(C)CCCC2)=O)O)CCN(C(c2ccc(O)nc2)=O)CC1 50695,C(CNC(=O)Cn1ncnn1)(CC(F)(F)F)NC(C(c1cccc(OC)c1)C)=O 50696,S(=O)(=O)(c1ccc(-c2ccc(C(C)N(C)C)cc2)s1)N(CC=C)CC 50697,c1(C(N2CCC(NC(c3c(SC)n(C)nc3)=O)C2)=O)c(C)cc(O)cc1C 50698,C1(OC)CC(N(C(=O)CCOC2CN(C(=O)CCc3cccnc3)C2)C)C1(C)C 50699,c1(CC(N2CCC(C(C)NC(=O)C(C)n3cnnn3)C2)=O)ccnc(Cl)c1 50700,C=C(C)CCCC(=O)N1CCC(C)C(CC(N2CC(CO)CC2CO)=O)C1 50701,c1(C(N2CC(C)C(NC(=O)CCCCC3CC3)C2)=O)ncc(C(F)(F)F)cc1Cl 50702,c1(N(CCc2ccc(C)cc2)C)nc2c(c(=NC3CCCSC3)[nH]1)CC(C)CC2 50703,C(=O)(CCCCCNC(N)=O)NC1(F)CN(C(CN2CC(C)(OC)C2)=O)C1 50704,C1(CCOC)CCN(C(=NCCc2ccnc(OC)c2)NCC2CCCCO2)C1 50705,N1(C(CC)=O)CC(=O)N2CCOCC2(CNC(=O)CC2CCCCC2(F)F)C1 50706,c1(CC)cccc(C(=O)NC(C(=O)NC2CN(C)NC2=O)C2CCCC2)c1 50707,C1(COC)(NC(=O)CCSC(F)(F)F)CCN(C(c2c[nH]nc2C(C)(C)C)=O)C1 50708,c1(CC(=O)NC(C2CN(C(c3ncccn3)=O)CC2O)C)csc2ccccc12 50709,C1(C)(C(N(C2CCCCCC2)C)=O)CC12CCN(C(=O)Cc1ncccn1)CC2 50710,c1(C(=O)NCC(O)CCNC(C2(CC)CCC2)=O)ccc(CN2CCCC2)cc1 50711,N1(C(CNC(CCC)=O)=O)CCN(C(=O)C(C)NC(C)(C)C)C(CC(C)(C)C)C1 50712,CCCCCC(F)C(=O)N1CCCC1(C(=O)NCC(C)C(=O)OC)CC 50713,Oc1nccc(=NC2CC(n3cnc4ccccc34)C2)[nH]1 50714,c1(OC)cc2c(cc1OC)C(NC(c1occ3c1CCC3)=O)CCCC2 50715,c1(OC)c(Cl)cc(C(N2CCC(NC(=O)CCC3CCC(=O)N3)C2)=O)cc1Cl 50716,N1(C(c2c(CC(N)=O)occ2)=O)CC2(CC(NC(=O)CN3CCCC3CO)C2)C1 50717,c1(N2CCC(CC#N)C2)nc(=NCc2nc(C(F)(F)F)cs2)[nH]c2c1CCCC2 50718,c1(CN2CCCCN(C)C(C)C2=O)c(F)cccc1F.C(C(F)C(=O)OC)OC 50719,CC(C)C(C)(C)C(=O)NC1COCC1NC(c1ccccc1OCCF)=O 50720,c1(C(N2CC3(C(NC(c4c(C)onc4)=O)CC3)C2)=O)cnc2cc(O)ccc2c1 50721,C1(C(=O)NC(C)CNC(=O)CCF)(CC)CCNC1=O 50722,c1(CCC)cc(C(=O)N(CCC(C)NC(=O)C(=C2CCCCC2)F)C)ccn1 50723,Cc1cccc(C(C)NC(=O)CCC2(C)CN(C(=O)CCC3(C)N=N3)C2)n1 50724,C(C(CO)C(C)(C)C)c1onc(-c2ncc(C)o2)n1 50725,C1(C(N(C)CC2CCCN(C(c3cn(C)nn3)=O)C2)=O)CCCC(F)(F)CC1 50726,C1(C)(C(N2CC(CC)(NC(c3ccc(C(F)(F)F)cn3)=O)C2)=O)COCC1(F)F 50727,S(=O)(=O)(c1nc(N2CCCC(F)C2)ccc1Br)N(C)CCOC(C)(C)C 50728,C1(NC(CN(C2CC2)CC)=O)CC2CC(NC(=O)Cc3cscn3)CC2C1 50729,N1(C(C(CC)(F)F)=O)CCC(F)(CNC(=O)CC2CCCC(C3CC3)O2)CC1 50730,C12(C(=O)OCc3cncc(C)n3)CCCC(CCC1)C2 50731,C(=O)(C(F)CC(CC)CC)NC(CC#C)(C)C(=O)NC1CC(C#N)C1 50732,O=C1CCC(C(=O)NC(Cn2cccn2)C(=O)NCCCCN2CCCC2)O1 50733,c1(OC)c(F)ccc(F)c1C(=O)NC1CCN(C(c2cc(C)ccn2)=O)CC1F 50734,C1(C(N2CCN(CC(C)NC(C3(C)CC3(C)C)=O)CC2)=O)Cc2cscc2C1 50735,N#CC1CN(Cc2cccc(C(N)=O)c2)CC1NC(c1ccc(O)c(O)c1)=O 50736,N1(C(c2ncn(C)n2)C(=O)N2CC(NC(N)=O)C2)CCC(O)C(F)C1 50737,Cc1ccccc1C(C)CC(=O)NC1CCN(C(=O)CCCF)C1 50738,N1(C(C2CCC(CNC(C3C(CC)CCO3)=O)O2)=O)CC(COC)C1(C)C 50739,C1(NC(C=Cc2scc(C)n2)=O)CC2CC(C1)N(C(=O)CC(C)C(F)(F)F)C2 50740,c1(SC)c(N2CCOC(c3cccc(OC(F)(F)F)c3)C2)nnc(Cl)c1C 50741,CCC(C)(C(=O)NCC(C)C(=O)Nc1conc1C)OC 50742,CC#CCCC(=O)NCCCCN(C(=O)COc1ccc(O)cc1)C 50743,Cc1cn(C)cc1C(=O)N(CC(C)NC(c1cc[nH]c1C)=O)C 50744,c1(C(N(CC(C)NC(C2(C)CC(F)C2)=O)C)=O)cn(C2CCOCC2)cn1 50745,CCC(C)(C(=O)N1CC(NC(=O)C(F)(F)c2cnn(C)c2)C(SC)C1)OC 50746,C1(NC(c2c(CC)scc2)=O)CC(NC(=O)C(C)C)C12CCOCC2 50747,N1(C(CCCOC)=O)CC(N=[N+]=[N-])CC1C(N1CCC(CF)C1)=O 50748,c1(OC)nc(Cl)ccc1C(=O)Nc1ncc(CCNCc2ccc(Cl)cc2F)s1 50749,c1(C2(C(=O)NC(c3ncc(Br)cn3)C)CNC2)cccc(F)c1 50750,N1(C(COc2ccc(OC)cc2)=O)CC(NC(=O)C(F)C2CCC2)CC(O)C1 50751,CC(C)CC(F)C(=O)NCC1(C)CCCN(C(c2c(Br)cnn2C)=O)C1 50752,N1(C(c2ncc(F)cn2)=O)CCCC2(CCO2)C1 50753,CC(CC(=O)NCC(C)NC(c1cnc(C(F)(F)F)s1)=O)C1CC1 50754,CCC(C)(COC)C(=O)NCC(C)N(C(=O)CC1CCC=CCC1)C 50755,N1(C(c2ccc3n[nH]cc3n2)=O)CCc2cc(Cl)c(F)cc21 50756,c1(C(=O)NCCCN(C(C2CCS(=O)(=O)N2)=O)CC)c[nH]c2ccc(Cl)cc12 50757,CCCCC(CNC(=O)CC1(OCC)CCC1)NC(=O)Cc1cccc(OC)c1 50758,CC1CCN(C(C2(C)CC2(C)C)=O)C1c1cn(CCS(C)(=O)=O)nn1 50759,CC1CN(C(=O)CCN(CCCO)C(C23CC(C#N)(C2)C3)=O)CC(=O)N1 50760,N1(C(Cc2cc(C)ns2)=O)CC2CC(NC(C3CC4CCC3CC4)=O)CC1C2 50761,N1(C(C(COC)O)=O)CC2CCCC(CNC(=O)CC3CCCC3)C2C1 50762,N1(C(Cc2cc(C)[nH]n2)=O)CCN(C(=O)CCN2CCSC(C)(C)C2)CC1CO 50763,N1(CC(=O)NCCC2(C)CC2)CCN(C(=O)Cc2cnoc2)CC1 50764,C(C)(CNC(C1CCCS1)=O)(CC(C)C)NC(CCOc1c(C)cccc1)=O 50765,C1(NC(CCCC#CC)=O)CCC(C)(C)CC1CNC(c1cnc(N)c(N)c1)=O 50766,C(C(=O)NCCCF)(C1=CCCCC1)N(CC)Cc1ccsc1Br 50767,C1(O)(c2cn(CC(=C)CC)nn2)CCN(C(=O)CCn2cccnc2=O)CC1 50768,C1(C(=O)NC(C)Cc2cccnc2)CC2CCC1N2C(C1(C#N)CCCC1)=O 50769,N1(C(C(C)OC(C)=O)=O)CCC(NC(C2CC(O)CN2C(N)=O)=O)C(C)C1 50770,S(=O)(=O)(c1ccc(N)c(NC(C2CCCC(COC)O2)=O)c1)NCC 50771,C1(CC(C)NC(C(COC)O)=O)CCN(C(c2cncc(F)c2)=O)CC1 50772,C=Cc1ccc(C(N2CCC(C)C(NC(=O)CCC(C)(C)F)C2)=O)cc1 50773,c1(C(=O)NCC(C)N(C)C(c2ccoc2Br)=O)c[nH]cc(Cl)c1=O 50774,N1(C(C2C(=C)C2)=O)CC2(CCNC(c3cc(N(C)C)cnc3O)=O)CCC1CC2 50775,C1(CC)CN(C(=O)C(F)=CCCF)CC1NC(c1cc(Cl)ccn1)=O 50776,C1(C(=O)NCCNC(CC(C)F)=O)CC(c2cccc(Br)c2)=NO1 50777,c1(C(N(C(CCNC(C2N(C(C)=O)CCOC2)=O)C)C)=O)nccc2n[nH]cc12 50778,c1(C(=O)NC2CC(C)(COC)N(C(c3cc[nH]n3)=O)C2)cnc(O)c2ccsc12 50779,n1(CC(CCSCC)C)nnnc1C(c1cnc(N(C)OC(C)=O)s1)OC 50780,Cc1c(C(=O)N(C2(C)CC2(C)C)C)cnn1-c1ccc(O)nn1 50781,c1(CC(=O)NC(C2CCCC2)CNC(CNC2CCC2)=O)cc(C)oc1C.CO 50782,C1(C(C)C)N(C(=O)CN2CCNC(=O)C2)CC12CC(N)C(O)C2 50783,CCS(=O)(=O)CC(=O)NC1CCCCC1NC(=O)C(C)=C1CCCC1 50784,N1(C(C2(C)COC2)=O)CCC2C1CCCN2C(=O)C(F)(F)c1ccccc1 50785,C1(F)(C(=O)NCC2CC(C#N)C2)CCN(C(=O)Cn2cncn2)C1 50786,CC1COc2c(C(N3CC(CCO)(NC(c4ccc(O)cc4)=O)C3)=O)cnn2C1 50787,C1(C)(NC(C(C)CC2CC2)=O)CCN(C(C2CC(C)(C)C2)=O)CC1 50788,Cc1sc(Cl)nc1C(N1CCN(C(C2CCCSC2)=O)CC1)=O 50789,N1(C(CN(C(C)C)C)=O)CCC2(NC(c3cc(F)ccc3N)=O)CC2C1 50790,C1(NC(C2CN(C(C)=O)C2)=O)CN(C(c2sc(F)cc2Br)=O)CCC1C 50791,C(C(C)C(F)C(=O)NCc1cccnc1O)NC(C1(CC#C)CC1)=O 50792,c1(NC(=O)Cc2cccc(-c3cn[nH]c3)n2)cc(Br)cnc1O 50793,c1(C(N2CC(C)N(C(C3CC34CCCC4)=O)CC2)=O)noc2ncccc12 50794,N1(N(C(=O)CCCn2cc(CCCN3CCOCC3)nn2)C)CCC(C)(C)C1 50795,N1(Cc2c(C)noc2)CCC2(NC(c3ccnn3CC3CCC3)=O)CCCC12 50796,C1(C)(OC)CCN(C(C2C=CC(NC(c3cccc(Br)c3F)=O)C2)=O)CC1 50797,N1(C(C=C(C)C(C)C)=O)CCCC12CCCN(C(=O)CC1(O)COC(C)(C)C1)C2 50798,c1(OC)ccc(C(=O)N(CCCCNC(=O)C(=O)N(C)C)C)nc1N 50799,c1(C(=O)NC2CN(C(c3cn(CC=C)nc3)=O)CC(C)C2)cc(C)c(=O)n(C)c1 50800,C1(CNC(C(C)Oc2ccc(F)nc2)=O)CN(C(=O)COCC2CC2)CCN1C 50801,N1(C(Cc2cccc(C)c2C)=O)CC2CCN(C(c3cn[nH]c3)=O)C2C1 50802,c1(C(=O)NCCC(C)N(C)C(c2ccnn2CC2CC2)=O)cc(C(F)F)ccn1 50803,c1(OC)cscc1C(=O)NC(C(N1CCCC1CN(C)C)=O)C1CCCC1 50804,c1(OC)ccc(CC(=O)NC2(C)CCCN(C(c3ccc(F)c(O)c3)=O)C2)cc1C 50805,C(=O)(CCC(CC)CCC)N1CC(O)(C(C(=O)NCc2cc(OCC)ncc2)F)C1 50806,C1(NC(c2cc(C)ncc2)=O)COCCN(C(=O)CNC(=O)NC2CC2)C1 50807,c1(CC(=O)N(C2CC(NC(=O)C=CCO)C2)C)ccc2c(c1)OCO2 50808,C(=O)(C1CCCc2n[nH]cc21)NC1COCCN(C(CCS(C)(=O)=O)=O)C1 50809,CC(C)(CCC(=O)NC1CCN(C(c2ccc(Cl)cc2)=O)C12CCC2)[N+](=O)[O-] 50810,C(=O)(C1=C(Cl)CCCC1)N(CC(=O)N(C1CCCC(C)(C)C1)C)C(C)C 50811,c1(SC)cc(C(N2CCC(NC(=O)C=CSCc3ccco3)C2)=O)ccn1 50812,CC(C)(CC(=O)N1CCC(NC(c2conc2C2CCC2)=O)C1)c1cccs1 50813,C1(O)(CC=C)CCN(C(=O)NCC2CCC2NC(=O)OC(C)(C)C)CC1 50814,c1(C(=O)NCC2N(C(C3(OCC)CCCOC3)=O)CC=C2)cc(NC)ccc1C 50815,Cc1c([N+](=O)[O-])c(C(=O)NCC(CO)NC(=O)CCCN(C)N=O)nn1C 50816,Cc1cc(C(=O)NC2CCCC(CNC(C3COC(=O)O3)=O)C2)n(C2CCC2)n1 50817,CC(O)CCCC(=O)NC(C1CCN(Cc2nc(-c3ccsc3)no2)CC1)C 50818,N1(C(c2coc(C(F)F)n2)=O)CCOCC(F)(CNC(C2C3CC4C(C3)C24)=O)C1 50819,CC(C)CCCCC(=O)NCC1CN(C(C2OCCC2C(F)(F)F)=O)CC1C 50820,N1(C(=O)CC2CCC(F)(F)C2)CCC(CCCCCn2cc(CO)nn2)CC1 50821,N1(C(C(CC)O)=O)CCC12CCCN(C(C1(Br)CC1)=O)C2 50822,C=C(C)c1cccc(NC(C2CCN(C(c3cscn3)=O)C23CCC3)=O)c1 50823,C(=O)(CCCCC(N)=O)NCC1(C)C(C)CN(C(C(C)OCC(C)C)=O)C1 50824,C1(CC)CCCCN1C(=O)C(CCN(C)C)NC(=O)C(CN(C)C)CC 50825,N1(C(C(C2CCCC2)OC)=O)CCN(C(c2cnc[nH]2)=O)C(C2CC2)C1 50826,c1(C(=O)NCCN(C(c2cnn(CCF)c2)=O)CC)cc2cccc(C)c2nn1 50827,C(C(C)C(C)C(=O)N(C)CC1(O)CCN(C(c2cn(C)cn2)=O)CC1)OC 50828,C(=O)(C1=CCC(F)(F)CC1)NC12CCN(C(c3ccc(C=C)cc3)=O)CC1C2 50829,C1(NC(C(c2cccs2)OC2CN(C(COC)=O)C2)=O)CC2(CCC2)C1O 50830,C(=O)(CCCC(C)(C)C)N1CCC(C)CC1CNC(=O)CCc1cccnc1Cl 50831,C1(NC(C(c2ccccc2)N(C)CC)=O)CN(C(=O)CNC(=O)OC)CCC1O 50832,N1(C(C2CC(CC)C2)C(=O)NCC2CCOC2)CC(OC)C2(CCCC2)C1 50833,CC(C)C(O)C(C)C(=O)NCC1CN(C(c2ccn(CCO)c(=O)c2)=O)C1 50834,CC1CN(C(c2cc(N(C)C)ccn2)=O)CCC1CNC(C1(CCF)CC1)=O 50835,n1(CC(=O)OC(C)(C)C)nccc1-c1cn(CCNC(c2cnc(Cl)[nH]2)=O)nn1 50836,C(=O)(CS(=O)(=O)C1CC1)NC1C2(CN(C(c3c(C)cc(O)nc3)=O)C2)CC1 50837,c1(CNCc2occ(C(=O)OC)c2C)c(C)ccc(F)c1N 50838,C1(C(=O)NC(C2(O)CCCCC2)C)(CO)CCN(C(C2CC(F)(F)C2)=O)C1 50839,C=C1CCN(C(C2CCN2C(C)(C)C)=O)C(C(=O)N(C(CCO)C(F)F)C)C1 50840,N1(C(=O)Cn2cc(C3CCCOC3)nn2)CCCC2(C1)C(O)CC2O 50841,N1(C(c2c(CC)ncc(Br)c2)=O)CC2CCC(C1)N(C(=O)C(C)C)C2 50842,Cc1cc(F)c(N)cc1C(N1CCN(C(c2csnn2)=O)CC1c1cn[nH]c1)=O 50843,N1(C(CNC(C)=O)=O)C(CC(N2CCC2C2CCCCC2)=O)C2CCCC12 50844,C1(C(=O)NC2CCN(C(=O)OC)CC2)CCC(C)(C)CC1 50845,N1(C(CCC=CC(C)C)=O)CC(CNC(C2CCC(CO)CC2)=O)C(C)C1 50846,CC(C(=O)NC1C2CN(C(=O)CCc3cccc(C(F)(F)F)c3)CC12)C(C)(F)F 50847,c1(C(=O)NCC2CC(NC(=O)C(=Cc3cccnc3)F)C2)ccc2nsnc2c1 50848,CCC(C)C(O)CC(=O)NC1C2CC(NC(C3(C#N)CC3)=O)CC12 50849,C1(CC)CN(C(=O)CN2CCC(O)CC2)CCN1C(=O)CNS(N)(=O)=O 50850,c1(C(=O)NC(CCNC(C(CC=C)C)=O)C)cnc2c(c1)N(C)CCO2 50851,c1(OC)ncccc1C(N1CCCC(CC(=O)NC(C)(C)CN2CCCC2)C1)=O 50852,CCC(CC)C(=O)NC(C)C(C)(C)NC(C1CC(=O)N(Cc2ccccn2)C1)=O 50853,C(CC(=O)N1CC(CN(C)C)C2(CC2)C1)(C(F)(F)F)NC(CSCC)=O 50854,N1(C(c2cc(C)n(C)c2C)=O)CC2COCCC2(NC(=O)COCC(F)(F)F)C1 50855,c1(C(N2CC(CNC(C3CC(OC)C3)=O)C(O)C2)=O)cc2cccnn2n1 50856,CCCCC(O)CC(=O)N1CC(C(=O)NC23CCC(CO)(CC2)C3)C(C)C1 50857,CCCC(CCCNC(c1cnc(OC)cn1)=O)NC(=O)CCc1cnc(C)o1 50858,Cc1ccc(C(N2CC(C(N3CCCC3C(F)(F)F)=O)C2)=O)c(O)c1 50859,C1(C(N2CC(OCC)C2)=O)CC(=O)N(C2CCNCC2)C1 50860,C1(NC(C(CC)N(CC)CC)=O)CCN(C(c2cc(C)cs2)=O)C(C)C1 50861,c1(C(N2CCC(N(C(=O)CN3CC4CC4C3)CCC)C2)=O)cc(N)c(O)c(F)c1 50862,CC1C(=O)N(CC2CCN(C(=O)NCC3(C4(O)CCC4)CC3)CC2)C(=O)C1C 50863,C(=O)(C(O)CCCNC(c1ccccc1C)=O)N(CC(CC)O)CC 50864,CC1(C)CCCC(C(=O)NC(CNC(=O)CCc2ncco2)C2CC2)C1 50865,c1(C(=O)NCCC(=C)CNC(C2(OC)CS(=O)(=O)C2)=O)ccc(C2CC2)nc1 50866,C=CCC(C(=O)NCCCN(C(=O)CC1CCC(C)(C)O1)CC)NC(C)=O 50867,C1(C(=O)NCC(c2ccccn2)C)CCC2(CC2)N1C(=O)C(C)CC(F)F 50868,CCCC(CCC)C(=O)NCC1CC2(CC2)CN1C(c1[nH]nc(OC)c1Cl)=O 50869,Cc1c(C(=O)NC2(C#N)CCN(C(c3ccon3)=O)C2)cncc1Br 50870,Cc1c(C(N2CCC(NC(=O)C=CC3CC3)C23CC3)=O)sc(Cl)c1Cl 50871,C1(C(=O)NCC(C(C)C)(C)F)CCCC(NC(C2CCCSC2C)=O)CC1 50872,N1(C(CCc2cc(C)on2)=O)CC(N(C(=O)Cc2nn(C)cc2Cl)C)C(F)C1 50873,C(=O)(C(CC(C)C)N(C)C)NCC(NOCC(=C)C)=O 50874,N1(C(CCCCCOCC)=O)CC(C(=O)OC)C2(C1)CN(c1ccncn1)C2 50875,N1(C(CCCSC)=O)CC(NC(=O)C(C)(O)C2CCC2)CC1C 50876,C1(NC(CC2(C#N)CCC2)=O)CCCCN(C(c2cnc(-c3ccsc3)s2)=O)C1 50877,C(=O)(C(O)C1=CCCCC1)N(CC(=O)NC(c1csnn1)C)C(C)C 50878,Cc1cc(Cl)nc(Cl)c1NC(C1CC(O)CCN1Cc1cc(F)c(Cl)cc1Cl)=O 50879,C1(C(N2CC(NC(CSc3ccc(C)cc3)=O)C2)=O)CC2CCC(C1)C2(F)F 50880,Cc1cc(C)c(C(N2CC=C(CNC(=O)CC3CCOC3(C)C)CC2)=O)cc1N 50881,N1(C(C2(C)C=CCC2)=O)CCN(C(c2onc3ccccc23)=O)CC(O)C1 50882,C(=O)(CC1CCCc2ccccc21)NC(CNC(C(CC#C)C)=O)(CC)CC 50883,c1(CNC(CCC)=O)cc2n(n1)CCN(C(C1(C)CC1(F)Cl)=O)C2 50884,CC(C)CC(Cc1ccccc1)CC(=O)N1CC(C)C(N)C1 50885,c1(CC(=O)NCC(C(=O)NC(CCC)C)N(C)C)ncccc1C 50886,c1(SC)nc(C(=O)NC2CC(C)N(C(=O)CC(=O)NCC3CC3)C2)cc(=N)[nH]1 50887,CS(=O)(=O)CCC(=O)NCCCC1CCCN1C(=O)CCc1cncc(F)c1 50888,N1(C(C(C)N(CC)CC)=O)CC(NC(C2CN(C(=O)N(C)C)C2)=O)C2(CCC2)C1 50889,c1(CC#N)ccc(C(=O)NC2CCC(NC(c3ccc(CF)cc3)=O)CC2)cc1 50890,C1(C(=O)NC2(CC=C)CN(c3nc4ccccc4o3)C2)CCc2nncn2C1 50891,C1(NC(C2(OCC)CCC2)=O)CC2CN(C(C3CSC3)=O)CC2C1 50892,Cc1c(CN(C(=O)CCCCN(C)C(c2ccncc2)=O)C)cnn1C 50893,C#CCCC(=O)N(CCC(=O)NC1CCOC1=O)CCCO 50894,Cc1ccc(NC(C2CCCC2CNC(c2ccc(CO)s2)=O)=O)c(C)n1 50895,C1(CCOC)(C(=O)NC2CC(O)(CNC(=O)C(C)C3CCC3)C2)CCCC1 50896,C12(C(=O)N(CCC3(NC(c4cc(CCC)on4)=O)CCC3)CC)CCCN1CCC2 50897,C(CCC(C)C(=O)NCCCCC(=O)NC1CCN(C)C1=O)OC 50898,Cc1c(Cl)sc(Cl)c1C(=O)NCC(C)N(C)C(c1cc(C(N)=O)c[nH]1)=O 50899,Cc1cc(C(=O)N(C2CC(C(=O)NCC3CC(O)C(O)C3)C2)C)cnc1O 50900,N1(C(C(C)(C)CCl)=O)CCOC2(CCN(C(=O)C(O)O)C2)C1 50901,Cc1cc(C(F)(F)F)nn1CC(=O)NCCC1CCN(C(c2cncs2)=O)C1 50902,N1(C(C(C)NC(C2CCCC2)=O)=O)CC(C)(C)CC1CNC(=O)CC1(C)CC1(F)Cl 50903,C1(CC)C(C(N2CCC2(C)CCO)=O)CCN1C(=O)Cc1cccnc1 50904,C1(CNC(C2(CC=C)CCCC2)=O)CN(C(=O)Cc2ccnc(O)c2)CCN1C 50905,C1(C2CCCO2)(C(=O)NCC2CC(C)N(C(c3ccncc3F)=O)C2)CCCO1 50906,C1(NCc2c(C)ncs2)CCN(C(=O)CC2(O)CCCC2)CC1C 50907,C(=O)(CC(=O)NC1(C(=O)NCCC(O)CO)CCCC1)OC(C)(C)C 50908,C(=O)(CC(O)C(=O)N1CC2CC2(CNC(c2coc(Cl)c2)=O)C1)OC(C)(C)C 50909,Cc1cnc(C(=O)NC2CC(F)CN(C(=O)C3=CCCCC3)C2)cc1C 50910,N1(C(CCC(C)(C)NC(=O)C=Cc2ccco2)=O)Cc2ccccc2C1 50911,C1(CCNC(CN(C)CCO)=O)CC(F)(F)CN1C(c1cccnn1)=O 50912,c1(C(=O)NCCCN(C)C)ccc2c(c1)CN(C(=O)C(=O)NCC(F)F)C2 50913,C1(NC(C(C)=C2CC2)=O)CN(C(c2nn(C)nc2C(F)(F)F)=O)CCC1C(F)(F)F 50914,C(=O)(CCCCCC(C)O)N1CCC(OCCNC(C(CC(C)C)O)=O)CC1 50915,C1(C(=O)NCCCCNC(c2cn(C)nc2O)=O)CS(=O)(=O)CC1C(F)(F)F 50916,C1(C#N)(C(=O)NC2(C)CN(C(CN(CC(=O)NC(C)C)C)=O)C2)CCCOC1 50917,CN1CC(C(N2CCC(F)(C(=O)NCCC(F)=C(F)F)C2)=O)CC1=O 50918,C1(NC(c2nc(C)n(C)c2)=O)CCCC(C(=O)N(CC(Cl)Cl)C)CC1 50919,CC1CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CCC1NC(=O)CC12CCC(CC1)CC2 50920,c1(CC(=O)NC2CCC2CNC(c2ccncc2)=O)ccc(F)cc1C(F)(F)F 50921,c1(CC)conc1CC(=O)NC(C(=O)NC1CN(CC2CC2)C1)c1cccs1 50922,CCC(CC)CC(F)C(=O)NCc1cc(C(=O)N(CC(O)C(F)(F)F)C)cs1 50923,c1(C(=O)OC(c2c(F)cccc2F)C2CCCC2)cnc(O)c2ccsc12 50924,C12CCC(CC1)NC2=O.C(=O)(C(C)=O)N(C1CCCC1)CC 50925,N1(C(C=C(C)Cl)=O)CCN(C(c2cc(S(N)(=O)=O)co2)=O)C(C)C1C 50926,C1(NC(CC(C2CC2)NC(C)=O)=O)CCCC(CNC(=O)C=C(C)C(C)(C)C)C1 50927,C(CC(C)C(=O)N(CCNC(c1cnc(O)o1)=O)C1CC1)=CCC 50928,C1(CCCC)CN(C(=O)C(CC(C)C)NC(N)=O)CCN1C(=O)C=CC(F)(F)F 50929,CC(CCNC(=O)C(C)Cc1ccco1)CCNC(=O)CCc1cn[nH]c1 50930,N1(C(c2ccc(CSCCC)o2)=O)CC2=C(C1)CN(C(=O)C=C1CCOCC1)C2 50931,C1(C(=O)NC(CC(=O)OC)C)CCCCCN1C(=O)CN1CCCC1=O 50932,C(C)(CN=c1ccn2ncc(S(=O)(=O)NCc3cc4ncccc4o3)c2[nH]1)OC 50933,c1(OC)cnc(C(N2CCCC(NC(=O)CC3CN(C)C3)CC2)=O)c(OC)n1 50934,C1(NC(CN(C)C(N)=O)=O)CC2(NC(C3CCN3S(C)(=O)=O)=O)COC1C2 50935,C(C)(C(=O)N(CCCCC(=O)NC1CC(=O)N(C2CC2)C1)C)(C(C)C)OC 50936,C#Cc1cc(C(=O)NC2CC(NC(=O)CCc3ccccc3C#N)C2)cc(F)c1 50937,CCC1=NOC(C(N2CC(C(O)C(=O)NCc3ccn(C)n3)C2)=O)C1 50938,c1(C(N2CC(CCCCNC(C3(O)CC4CCC3C4)=O)C2)=O)cc2sccc2s1 50939,C1(OC)CC(NC(c2cc(C)nn2C)=O)C12CCN(C(c1scnc1C)=O)CC2 50940,c1(OC)cc(C(=O)Nc2ncc(-c3ccc(C)nc3F)cc2C)ccc1F 50941,CC1(NC(=O)CC2CC(F)C2)CCC(NC(c2ncoc2C(C)(C)C)=O)CC1 50942,CC1CC(CNC(=O)CCCc2cnn[nH]2)CCN1C(=O)CC1CCCO1 50943,c1(C(=O)NCCC2CCN(C(=O)C=Cc3cnc[nH]3)C2)coc2c1CSC2 50944,c1(C(=O)NCC2CC2NC(C2CCC2)=O)ccc2nc(O)nc(O)c2c1 50945,N1(C(C(COC)OC)=O)CCC(CCC(C)(C)NC(c2cnc(S)[nH]2)=O)CC1 50946,C1(NC(NC(COC)C)=NCCCNS(C)(=O)=O)CCS(=O)(=O)C(C)(C)C1 50947,N1(C(CCSC)=O)CCCCC(NC(=O)CC(C(C)C)c2ccccc2)C1 50948,Cc1cc(C(=O)NC2CN(C(c3cccc(O)c3C)=O)CC2C)c2n[nH]cc2c1 50949,Cc1c(O)ccc(CNC(C2(Cc3coc(C#N)c3)CCC2)=O)c1O 50950,O=C(CC(C(F)(F)F)NC(=O)C(c1ccccc1)OCC1(C2CCC2)CC1)OC 50951,N1(C(CC(C=C)(C)C)=O)CCN(C(=O)CCCN(C)C)C(C)C1C 50952,C(=O)(C(C(C)CC)NC(c1ccc(SC)o1)=O)NCCSCCC=C 50953,c1(CC)c(C(=O)NC(CNC(=O)COCC2CCCO2)CC2CC2)cccc1F 50954,CN1CCC(C(=O)NC2CC(F)CN(C(C3CCC3C#N)=O)C2)CC1=O 50955,Cc1cnc(NCC2CCCCC2NC(C2(O)CCOCC2)=O)nc1O 50956,Cc1cc2ccc(C(=O)NC3CCCN(C(c4ccc(=N)[nH]n4)=O)CC3)cn2c1 50957,N1(C(COCc2cccc(C)c2)=O)CCC(NC(=O)CCOC2COC2)C(O)C1 50958,N1(C(c2c(C)[nH]cc2)=O)CCC(O)(CCNC(C2(C3CCCCO3)CC2)=O)CC1 50959,CC(C)C(C)C(CNC(=O)C=Cc1ccoc1)NC(=O)CCCCCN(C)C 50960,c1(C(=O)NC(CCNC(C(CCCC)CC)=O)C)cccc([N+](=O)[O-])c1OC 50961,CC(C)C(C(=O)NC12CC1CN(C(=O)CCCNc1cccs1)C2)NS(N)(=O)=O 50962,C1(NC(COc2cc(C)on2)=O)CC2CN(C(=O)C3=CCCO3)CC12 50963,C1(C(=O)NC(C)C(C)NC(C2CC(Cl)(Cl)C2)=O)CCCCC(=O)N1 50964,C12(COC)CC(CNC(C3CC3C3CCCO3)=O)(CN1C(c1cnn(C)c1)=O)C2 50965,C1(C2CCOCC2)(C(=O)NC2CC(NC(C(C(C)C)OCC(C)C)=O)CC2O)CC1 50966,C(=O)(C(CN(C)C)C(C)C)NCC(C1N(C(c2[nH]cc(C)c2)=O)CCC1)(C)C 50967,C=C1CCN(C(c2nonc2N)=O)C(C(=O)Nc2cnc(F)nc2)C1 50968,C(=O)(CC1=CCCC1)OC(C(C(=O)OCC)=O)C 50969,c1(C(N2CCC(N(C(c3cscc3OC)=O)CC)C2)=O)oc(C)nc1C 50970,CS(=O)(=O)C(CNC(=O)Cc1cccc(Cl)c1)CNC(c1cc(C#N)cs1)=O 50971,c1(OC)cccc(NC(c2sccc2CNC(=O)N(C(C)C(=O)OC)C)=O)c1 50972,N1(C(C(C)=C2CCC2)=O)CCC(NC(c2cc(C(C)(F)F)ccn2)=O)CC1C 50973,C(C(=O)N1CCCN1)NC(C1CC2CCC1C2)=O 50974,CC1CCN(C(=O)CCc2cncnc2)CCN1C(c1cccc(N(C)C)n1)=O 50975,N1(C(c2ccc(C(C)C)o2)=O)CCC(O)(C2CCN(C(c3cnns3)=O)CC2)C1 50976,N1(C(C2CN(C(CCNC(=O)CO)=O)CC23CCC3)=O)CC2CCC(O)C(O)C12 50977,C(C(C)(CC(C)C)NC(c1csnn1)=O)NC(c1c(C)cc(C(F)(F)F)s1)=O 50978,C1(CNC(C(C)(C)NC(C)=O)=O)CCN(C(=O)Cc2ccc(O)c(Cl)c2)CC1(F)F 50979,C1(CNC(c2ccc(C(C)C)cn2)=O)CCC2(CCC2)C1NC(=O)C=C1CCC1 50980,CC(C)CC(CNC=O)CC(=O)NC1CCCN(C(=O)C=CCN2CCCC2)C1 50981,N1(C(c2c(C)nc[nH]2)=O)CC(C)C(NC(=O)C=CCO)C(C)C1 50982,c1(C(=O)NC2(C3N(C(COC)=O)CCC3)CC2)ccc(OCC(C)(C)C)cc1F 50983,C(=O)(C1COc2ccc(Cl)cc21)N1CCC(CN(C)C(C2CC3CC3C2)=O)C1 50984,c1(C(N2C(C)(CNC(c3cnc(SC)[nH]3)=O)CCC2)=O)cccc(N)c1O 50985,C(=O)(C(F)(CNC(=O)C(C#N)C(C)(C)C)C(C)C)N(CC(C1CC1)OC)C 50986,CC(C)C(F)C(=O)NCC1CCC(NC(=O)CC2CC(C(F)F)C2)C1 50987,N1(C(c2cn(C)c(=O)cn2)=O)CCC(NC(=O)CNS(N)(=O)=O)CC(O)C1 50988,C1(N(C(=O)CSc2cccs2)C)CCCC(NC(c2c[nH]cc2Br)=O)C1 50989,C1(NC(C(COC)O)=O)CN(C(=O)Cc2cccs2)CC1S(C)(=O)=O 50990,c1(C(=O)NCC(C(C)C)NC(C2COCCO2)=O)sc(N2CCOCC2)nc1Cl 50991,c1(OCC(=O)N(C2CCN(C(C34CC(O)C3C4)=O)C2)CC)cc(Cl)ccc1Cl 50992,C=Cc1ccc(C(=O)NC(C2(O)CCN(C(=O)CSc3nncs3)C2)C)cc1 50993,c1(C(=O)NC23CCN(C(=O)C(N4CCOCC4)O)CC2C3)ccc(Cl)cc1Cl 50994,N1(S(CC(=O)OCC)(=O)=O)CC2(CCN(S(=O)(=O)c3cnc(OC)s3)C2)C1 50995,c1(OC)cc(CN2CCNCC2)ccc1I.c12ccc(nc1)[nH]2 50996,c1(C(=O)NC2(C)CN(C(C3(CC(C)C)CCC3)=O)C2)nn(C)c2ccccc12 50997,CCC(C)C(C)C(=O)NCc1ccc(NC(=O)OCC)cc1.C12CCN(C1)C2=O 50998,c1(C(N2CC(O)(C(C)NC(CNC(=O)OCC)=O)C2)=O)cnc2c(c1)CCOC2 50999,Cc1ccc(C(=O)NC2CCN(C(=O)C(C)N(C)C)CC2(C)C)cc1[N+](=O)[O-] 51000,NS(=O)(=O)c1ccc(C(N2CCOCC2C2CCCCCC2O)=O)c2nsnc12 51001,C1(CC(=O)NC2CN(C(=O)CCCc3cccc(F)c3)C2)(CSC)CCCCC1 51002,c1(C(N2CCN(C(=O)Cc3nc[nH]n3)C(CO)C2)=O)nc(Br)c2n1CCCC2 51003,C1(C(=O)NCCC(=O)NCC)CC2(CCN1C(c1cn(C)nn1)=O)CC2 51004,C1(NCCN(C(=O)COCCN(C(=O)CSC(F)F)C(C)C)C)CCCCCC1 51005,c1(-c2cn(CCNC(c3cc(COC)[nH]n3)=O)nn2)cc([N+](=O)[O-])ccc1OC 51006,O=C1CN(C(c2ccnc(Br)c2F)=O)CCN1Cc1ccc(F)cc1F 51007,N1(C(C(C)SCC)=O)CCOCCC1C(N1CC(C2CCN(C)CC2)C1)=O 51008,CCCC(C(=O)OC)C(=O)NC1COCCC1NC(c1ccc2n[nH]cc2n1)=O 51009,c1(C(N2CCCC(NC(CCOCCOC)=O)C2C)=O)cc2c(s1)CCC(C)C2 51010,CCCCC(O)CC(=O)NC(CC(F)F)C(=O)N1CCOC2CC12 51011,N1(C(c2c(CC)csc2)=O)C(C(=O)NCCOC(C)=O)CCC12CC2 51012,C1(CNC(c2cc(C3CCC3)no2)=O)CN(C(C2(CO)CCCC2)=O)CC1(F)F 51013,c1(OCCC)ccc(Cl)cc1NC(N1CCC(C)C1(C)C)=O 51014,CC1CN(C(C(=O)NCC2CC2)C(C)CC2CCOCC2)CC(C)(C)C1 51015,c1(OCC)ccccc1NC(C(c1c(C)n[nH]c1)N1CCC(CC(F)F)C1)=O.OC 51016,C1(NC(CCc2cc(C)no2)=O)(CO)CCCN(C(C2CC23CC(C)(C)C3)=O)C1 51017,N#CC1(C(=O)NCCc2ccc(Br)cn2)CC12CCCC2 51018,N1(C(CNC(=O)NC)=O)CCN(C(CNC(=O)C=CC2CCCC2)C(F)F)CC1 51019,c1(C(C(=O)NCCCF)N(CCC#N)CC)ncc(Cl)cc1Cl 51020,N1(C(c2ncn(CC)c2)=O)CCN(C(=O)C(F)(F)C(F)F)CC1CO 51021,N1(C(c2n(C)cnc2)=O)CCCC2(CCC(NC(c3coc(Cl)n3)=O)C2)C1 51022,C=C(C)CC(C(=O)NC(CNC(=O)CN1CCOCC1=O)CCC)NC(C)=O 51023,CC1CN(C(=O)C(C)Cn2cccn2)CC(C(=O)NC(C2CCCO2)(C)C)O1 51024,C1(CC)CN(C(C2(NC(=O)C(CC3CCC3)OC)CCOCC2)=O)CCO1 51025,C(CC(=O)N1CC(F)(F)C1C1CC1)(C(F)F)NC(c1n(C)c(S)nn1)=O 51026,CCCS(=O)(=O)CC(=O)NC1CN(C(c2ccc(O)nc2)=O)CC1CO 51027,c1(OC)ccc(CC(N2CC(NC(=O)CC3CC(OC)C3(C)C)C(O)C2)=O)cc1 51028,c1(C(=O)NCC(F)CNC(C2CC(F)C(=O)N2)=O)cc2cccc(O)c2[nH]1 51029,c1(N2CC3C(NC(c4ccc(S)cc4)=O)C3C2)ncnn2cccc12 51030,C(=O)(C(C)S(=O)CCCc1nc2ccccc2n1C)N(CCCC)C 51031,C=C1CC(CN(C(C(=O)OC)C2CN(C(=O)NC(C)(C)CC)C2)C)C1 51032,CCCS(=N)(=O)c1cccc(CNc2cccc(C#N)c2F)c1 51033,C=CC(CC)CC(=O)N(CCCNC(C12CCN(CC1)C2)=O)C1CC1 51034,C=C(C)CCCC(=O)N1CC=CC(NC(C2(Cc3cccc(F)c3)CC2)=O)C1 51035,C1(C(N2C(C)CCC(NC(CN(CCOC)C)=O)C2)=O)CC2(C1)CC1(CCC1)C2 51036,CC1(C)CN(C(c2ncccc2C(F)F)=O)CCC1NC(=O)CC1CCC(=O)N1 51037,c1(C(=O)NCC(C)N(C(COCCCCC)=O)C)[nH]c(C)cc1C 51038,N1(C(C(C#C)(C)C)=O)CCN(C(=O)CC2CCNC2=O)C(CC(F)(F)F)C1 51039,C(C(COC)C(=O)NC1CC(C(=O)NC2CC(OC)C2(C)C)C1)OC 51040,C(C(=O)NCCCCC(=O)NC(C12CC(CO1)C2)C)(C(C)C)OC 51041,Cc1cc(C(=O)N(CC(C)N(C(=O)C(c2cccs2)N(C)C)C)C)c(N)c(C)c1 51042,CC1CC(NC(=O)CCc2cnn[nH]2)CN1c1nnco1 51043,c1(CC)ccc(C(=O)N(CC(C)NC(=O)Cc2ccsn2)CC)cc1 51044,C1(O)(CC(=O)NCC(C(=O)NC2C(CN(C)C)CCC2)O)CCCCC1 51045,CC1(C)C(NC(=O)C(CC2CCCC2)CN)C(C)(C)C1O 51046,C=CC(CC(=O)NC1(CNC(=O)COCC)CCCC1)c1ccccc1 51047,Cc1ccnn1C(C)C(=O)NC1CCCCC1.C12CC(C1)CNC2=O 51048,c1cn2c(n1)C(Nc1cc(NC3CCN(c4ccncn4)CC3)ncn1)CCC2 51049,N1(C(c2cn(C3CC3)nn2)=O)CCN(C(=O)CN2CCCS2(=O)=O)C2CCC12 51050,C(CC)(C(=O)NC(C1CN(C(=O)CC2CC2C)C1)C)=CC 51051,N1(C(c2c(C)noc2N)=O)CCN(C(C2CCC(=O)N(C(C)C)C2)=O)C(C)C1 51052,c1(OC)cccc2c1CCCC2Nc1cc(N2CCC(CN3CCCC3)C2)ncn1 51053,c1(NC2CC(NC(C3C(OCC)C3C)=O)C2)ncc(C(N)=O)cc1Cl 51054,c1(C(=O)NCC(CC(C)C)NC(CC2CC(CC)C2)=O)c(F)cncc1Br 51055,c1(C(=O)NCC2CCN(C(C(CC=CC)C)=O)C(C)C2)cn2ccccc2n1 51056,c1(C(c2ccccc2)NC(CC)C2CC2)ccccc1Br 51057,C1(C(C)C)CN(C(C2CNC(=O)C2)=O)CCN1C(=O)CCc1cnc[nH]1 51058,c1(CCCC(=O)NCC2CC(OC)CN2C(=O)C(F)F)c(F)cccc1F 51059,N1(C(COCCC)=O)CCN(C(=O)CCc2cc(C)n(C)n2)CC2(CC2)C1 51060,CCCCCCC(CC)(c1nnnn1CCOC)NCc1ccc([N+](=O)[O-])o1 51061,N1(C(C(C)(C)c2cncnc2)=O)CCC(CNC(=O)C(=O)Nc2ncc[nH]2)CC1 51062,C(Nn1cncn1)c1cn(C(F)F)nc1.O(C(F)(F)F)CC 51063,c1(C(N2C(C(=O)Nc3ncc(F)s3)CC(F)C2)=O)c(F)cccc1F 51064,C1(C(=O)NCC2(C)CCN(C(c3cnco3)=O)C2)(CC)CNC(=O)C1 51065,c1(C(=O)NC2CN(C(c3nc(C)nn3C)=O)CC2C)cnn2ccn(C)c12 51066,Cc1cccc(C(=O)C(=O)NCC=CCNC(=O)CN(C)CCO)c1 51067,C#CC(N(C)N(C)Cc1ccc(-c2ccc(F)cc2)cc1)C1CC1 51068,Cn1cc(S(N)(=O)=O)c(C(=O)NC2CC(C)(NC(=O)CC3CCC(=O)N3)C2)n1 51069,CC(C)(C)C(CO)C(=O)N1CC2CC1CN2C(=O)CCCC1CCCO1 51070,CCCC(C)(CC)C(=O)NCC(C1CCC1)NC(c1cnc(OCC)c(Cl)c1)=O 51071,N1(Cc2nnc(CC)s2)C2CCC1CN(C(c1cc(C)[nH]n1)=O)CC2 51072,Cc1c(C(=O)N(C)CCOCCCNC(C2(O)CC(F)(F)C2)=O)cccc1F 51073,N1(C(C(C2CCCC2)OC)=O)CC(=O)NCC1C(=O)NCCC(F)=C(F)F 51074,N1(C(CC(=C)C)=O)CCN(C(=O)COc2ccccc2C#N)CC1C1CC1 51075,C1(C(=O)NC2(CC=C)CCN(c3ncccc3C(C)=O)C2)CCOC2(CCC2)C1 51076,c1(OCC)ccc2c(c1)CCN(c1nc(O)c3cnn(C)c3n1)C2 51077,C=CCC(C)(O)C(=O)NCCC(=O)NC1CC(O)C1(C)C 51078,CCCC(CCC)C(=O)NCC1CC1C(N1CCC(OC)C1(C)C)=O 51079,c1(C(N(CC(CC)NC(c2c(OCC)cccn2)=O)C)=O)c(OC)cccc1C 51080,c1(CC)c(C(=O)NC(CNC(c2ccsc2C(F)F)=O)CO)[nH]c(C)c1C(C)=O 51081,C(C)(C)(CCC(=O)NC(C)C)NC(C1(OC)CCC(C)C1)=O.C(CC(=O)O)N 51082,C1(CC)CC(C(=O)N(C2CCC2C)C)CCN1C(c1nn(C)cc1Cl)=O 51083,N1(C(C2=NOC(C)C2)=O)CCC(C2(NC(=O)C=Cc3nccs3)CC2)C1 51084,C1(OC)CN(C)CC1NC(=O)C(C1CCCC1)NC(C1CC1(C)C(F)F)=O 51085,c1(C(C(=O)NCCN(CC)CC)N(C)CCC2CCCO2)ccc(F)c(Br)n1 51086,C(=O)(CCCC(C)=O)NCC(CC=C)NC(=O)C=Cc1ccco1 51087,CC1(C)CCCC(C(=O)NCCC(C)(C)NC(C2C3CCCCC23)=O)C1 51088,C1(C(N2CC(N(C)C3CC3)C2)=O)(COC)C=CCN1C(C1C2CCCOC12)=O 51089,C(=O)(C(CC)C(C)C)N1CC(C=C)(C(=O)NC(CO)CC=CC)C1 51090,N1(C(C(COC(C)=O)C)=O)CCC(C(=O)NCCNC(=O)C(C)C)CC1(C)C 51091,N1(C(C=CC(C)(C)SC)=O)CCN(C(=O)CCNC2CCCC2)C(CF)C1 51092,CCCC(C(=O)N(CCCN(C(=O)CCc1cc(C)sc1C)C)C)NC(N)=O 51093,Cc1nn(C)c2[nH]c(=NCCC3(CNC(C4CC4(C)Br)=O)CC3)c(C#N)cc12 51094,CC1COCCC1NC(=O)C(=O)N(CCCC1CC2CCC1C2)C 51095,CN1CCC(CCNC(=O)CC2C=CC(NC(c3cncn3C)=O)C2)C1 51096,Cc1cc(CC(N2CC(NC(=O)C(C)(C)C3CCCC3)C(CO)C2)=O)ccn1 51097,C12(C(=O)NCC3C(C)(C)N(C(C4CCCOCC4)=O)CC3)CCC(N=[N+]=[N-])C1C2 51098,Cn1nnc2cc(C(N3CCC(CCNC(C4CCCC(F)(F)C4)=O)C3)=O)sc12 51099,C1(NC(c2c(CC)noc2C)=O)C2CCN(C(c3ccoc3)=O)CC12.C1(=O)CN1 51100,c1(SCC)ccc(C(=O)NCC(CCCC)NC(C2CSCCS2)=O)cn1 51101,C1(C(N(CCCNC(C(n2ccc(C)n2)(C)C)=O)C2CC2)=O)C(Cl)(Cl)C12CC2 51102,N1(C(C=COCC)=O)CC(NC(=O)CCC2CCCCN2C)CC(C)(C)C1 51103,C(=O)(CCCCCCC(=O)OC)NC1CN(C(CCC(=C)C)=O)CC(F)C1 51104,Cc1ncc(C(=O)N(C)CC2(NC(=O)C3=COCCC3)CC2)c(Br)c1Cl 51105,Cc1cccc2c1OC(C(=O)NC1CN(C(c3ccon3)=O)CC1C)C2 51106,C1(C(N(CCNC(c2ccc(OC(C)C)nc2)=O)CC)=O)CCC(F)(F)C1O 51107,C(CN=C(NCCn1cccn1)NCC1CCNC(=O)C1)c1ccc(OC)cc1 51108,C1(NC(Cc2c(C)ccc(F)c2)=O)CCCC12CN(C(C1NC(=O)C3CC13)=O)C2 51109,CC(CC(=O)N1CCN(C(=O)C=C2CCOCC2)CC1)C(C)(C)C 51110,c1(C(=O)NCC2(OC)CN(C(c3nocc3C)=O)C2)n[nH]c(C(C)C)c1Br 51111,NS(=O)(=O)c1n[nH]cc1C(N1CC2CCC1C2NC(=O)Cn1cnccc1=O)=O 51112,CCCC(CCC)C(=O)NCc1occc1C(=O)NC1CCOC1C1CC1 51113,c1(C(=O)NC2CN(C(c3ccc(C(C)C)o3)=O)C3C2C3)cc(F)cc(F)c1 51114,c1(OC)ccncc1C(=O)NC1CCN(C(C2CC2C)=O)C1C 51115,c1(C(=O)NC(CNC(C2C(C)CC2)=O)(C)C)ccc(C(F)F)cc1Cl 51116,C(CN=c1ccc(Br)c(S(=O)(=O)NCc2c(F)cc(Br)cc2F)[nH]1)C1(C)CC1 51117,Cc1ccc(C(C)NC(C2CC(O)(CNC(=O)OC(C)(C)C)C2)=O)c(Cl)c1.C 51118,CC1CN(C(C2C(F)(F)C23CCC3)=O)CCC1CNC(=O)CC1OCCC1(C)C 51119,C1(OC)CCC(C(=O)NC(C)CNC(c2sccc2C(C)(C)C)=O)CC1 51120,C(C)(C)(C(=O)NCCCC1(NC(=O)CC2CC(F)C2)CC1)OCC 51121,C1(C(=O)NC(c2n(C)ncc2)C(=O)NC2CC(O)C2)C2CC3C(C2=O)C13 51122,CC1OCCC1(O)CNC(C1(NC(C2CNC(=O)N2)=O)CCCCC1)=O 51123,N1(C(CN2CCC(C)C2)=O)CC2CCC1CN2C(=O)C(C1CCCCC1)O 51124,CCCCCC(=O)NC1CN(C(c2cnn(C(C)C)c2C)=O)C2CC12 51125,CC1CN(C(c2ccn(CCN(C)C)n2)=O)CC(C)N(C(=O)C(C)C2CC2)C1 51126,c1(C(C(=O)NCC=C)N(C2CCN(CC)C2)CC)cnn(C)c1Br 51127,C(=O)(C1CCc2c[nH]nc21)N1CCC(C(C)NC(c2cnsc2)=O)CC1 51128,C1(CC(=O)NCCc2nc(=N)[nH][nH]2)NC2CCCC12 51129,C#CCC(CC#C)C(=O)NCC(CO)NC(=O)CNC(=O)Nc1ccccc1C 51130,CC(C(=O)N1CC(NC(C2CNC(=O)N2)=O)C(C)C1)C(C)c1ccccc1 51131,c1(CCCC)ccc(C(c2nnnn2C)NCCc2csc(C)n2)cc1 51132,C(C(=O)NCC1(NC(c2c(Cl)cnn2C)=O)CCC1)(C(C)C)SC 51133,C1(C2CCN(C(C3(C)CC3C(F)(F)F)=O)CC2)(C(=O)OC)CC(F)(F)C1 51134,N1(C(=O)NCC2(COC)CCCC2)CCN(c2cccc(F)c2)C(=O)C1 51135,c1(C(N2CC(CNC(c3ccc(SC)cc3)=O)C3C2C3)=O)cncc(Cl)c1C 51136,Cc1ccc2c(c1)C(C(=O)N1CC(CNC(=O)CCOC(C)CC(C)C)C1)CC2 51137,CC1CN(C(c2ccns2)=O)CCCN1C(=O)CCc1cccc(OC(F)F)c1 51138,N1(C(CC(C)C(F)F)=O)CCC2CCCC12C(=O)NC(C1CCC1)C1CC1 51139,CCC(F)(F)C(C)(C)C(=O)N1CC2CC1CN2C(c1ccc2oc(C)nc2c1)=O 51140,c1(-n2ccc(C(N3CC4(CCC4O)C3)=O)n2)ccc(O)cc1Cl 51141,C12(C(N3CC(C)(NC(c4ncc(OCC)nc4)=O)C3)=O)CCCCC1OCC2 51142,C#CC1CC2CCC1N(C(C1CCN(C(=O)CCC3CCCN3C)C13CC3)=O)C2 51143,Cc1nc(C(F)F)cc(N2CCOC(CCF)C2)n1.C1(N)CCCCC1 51144,c1(C(N2CC(OC)(CNC(c3cnnn3C)=O)C2)=O)cc2ccccc2[nH]1 51145,c1(C(N(CC)CC2CCCN2C(C2OCCC2C(C)C)=O)=O)cccc(=S)n1O 51146,CC(C)(C(=O)NCCN(C1CCCC1)C(C1OCCOC1C(F)(F)F)=O)C(N)=O 51147,N1(C(CCC=C)=O)CCN(C(=O)C(c2ccccc2F)C)CC1CCO 51148,CCC(C)(COC)C(=O)N1CC(C2CC2C(N2CCOC(CCO)C2)=O)C1 51149,N1(C(CCP(C)(C)=O)=O)CC(CNC(=O)Cc2cccc(C#N)c2)CC12CCC2 51150,c1(OC)ccc(Cl)cc1CC(=O)N(C1CC(NC(=O)CC2(O)CCCC2)C1)C 51151,c1(NC(C2CCN(C(c3cc(C)nnc3C)=O)C2C)=O)cccc2c1CCO2 51152,C1(SC)CN(C(c2oc(CO)cc2C)=O)CC1NC(c1ccsc1SC)=O 51153,N1(C(CCC)=O)CCN(C(c2cc(C)nn2C)=O)C(CCO)C1 51154,C1(C(=O)NCC(CNC(=O)CN2CCS(=O)(=O)CC2)O)CC2C=CC1C21CC1 51155,c1(C(N2CCC(CNC(C(CC)O)=O)C2)=O)cc2ccccc2c(=O)n1C 51156,CC1CCN(C(C2CNC(=O)O2)=O)CCN1C(c1ccnn1CCF)=O 51157,N1(C(c2ccc(C(CC)=O)cc2)=O)CCN(C(c2coc(C)n2)=O)CC1C1CC1 51158,Cc1ccc(C(=O)NCCSCC(=O)NCC(C)(C)O)c(F)c1 51159,c1(C(N2C(CN(C(=O)Cn3nnc(C)n3)CC)CCC2)=O)cc(C)nc(O)n1 51160,N1(C(c2c(C)snn2)=O)CCCC(C(C)C(=O)Nc2ccc(Cl)cc2)C1 51161,C1(C#N)(C(N(CC(C(=O)NC(CCOC)CO)C)C)=O)CCCOC1 51162,N1(C(C(C)(C)C)=O)CCC2CCCC12C(=O)NCCC1(N(C(=O)CCF)CC)CC1 51163,CCC(C)(C)CC(=O)N1CC(N(C(=O)C(C)OC)C)C(O)C1 51164,C1(CNC(C=CCC)=O)CN(C(=O)C(=O)NCCOC)CCC1C 51165,N1(C(C2C(CCOC)C2)=O)CCCN(C(=O)Cc2sc(S)nc2C)CC1C 51166,N1(C(C2C(NC(C(CC3CC3)OC)=O)CC=CC2)=O)CC(C)N(C)C(C)C1 51167,N1(C(CNS(CCCC)(=O)=O)=O)CCc2nc[nH]c2C12CCN(C(=O)C(N)=O)C2 51168,c1(NC(=O)NCC=CCCOC)cnc2ccccn2c1=O 51169,Cc1ccc(C)c(C(=O)NC(c2ccccc2)C(C)NC(c2ccncc2)=O)n1 51170,c1(C(C(=O)NCCCC(C)NC(C(C)NC(C)=O)=O)(C)C)ccc(F)cc1 51171,C1(C(=O)NC(C)Cn2cc(C3(N(C)C)CCC3)nn2)CCC(N(C)C)CC1 51172,c1(NC2CC(C)N(C(c3cc([N+](=O)[O-])c[nH]3)=O)CC2)ncc2c(c1C#N)CCC2 51173,C1(OC)(CNC2(c3ccccc3)CCC2)CCCS(=O)(=O)C1 51174,c1(C(N2CC(CNC(C(C)c3ccsc3)=O)C2)=O)ccc(-c2ccco2)o1 51175,N1(C(C2ON=C(C(C)C)C2)=O)CCC(N=[N+]=[N-])(C(=O)Nc2cc(O)cc(F)c2)C1 51176,Cc1cc(O)ncc1C(=O)N(CCCN(C(=O)CC1CCC(=O)N1)C)C 51177,N1(C(=O)COc2c(F)cccc2F)CC2(COC(CNC)C2)C1 51178,Cc1cnc(C=CC(=O)NCC2(NC(C3CC(F)(F)C3)=O)CCOC2)[nH]1 51179,N1(C(=O)Nc2cn(C(=O)OC(C)(C)C)nc2)Cc2ccccc2OC(C)C1 51180,C1(CC=C)CCCN(C(=O)CCC2(C)CCN(C(C3(n4cccn4)CC3)=O)C2)C1 51181,Cc1ccc(C(=O)NC(C)CN(C(=O)C(C(C)O)N(C)C)C)cc1I 51182,c1(C(C)C)cc(C(=O)NC2CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)C2)cc(Br)c1 51183,C1(NC(=O)C=CBr)CN(C(=O)COc2ccsn2)CC(F)(F)C1 51184,CC(C)(CCNC(C1OCC1(C)C)=O)NC(=O)CNC(c1ccccc1)=O 51185,C1(C2(O)CCC2)(C(=O)NC(C)C(CO)NC(C2CC3CC2CC3O)=O)CC1 51186,c1(CC)cnc(C(=O)NCC2(NC(C3CCC34CCC4)=O)CCCC2)cn1 51187,N1(C(=O)C(c2cccnc2)O)CC2CC(C(N3CCCC4CC34)=O)(C2)C1 51188,c1(C(N2C3C(NC(C(C(CC)CC)C)=O)C(C3)C2)=O)nc(N)cc2ccccc12 51189,N1(C(C(CC)(F)F)=O)CCC(C)C(N(C(=O)COCc2ccccc2)C)C1 51190,C1(NCC2CCCN(C(Cc3c(C)cccc3)C)C2)CCC2CC2CC1 51191,C1(CSC)(NC(c2cc(Br)ccn2)c2nnnn2C)CCOCC1 51192,C1(NC(C(CC#C)O)=O)C2CCN(C(C3(C4CC4)CCCO3)=O)CC12 51193,c1(OCCC(=O)NC(C)C(c2ccccc2)N)ccc(C(F)(F)F)cn1 51194,CC1(C)CN=C(N2CCN(Cc3ccccc3S(C)(=O)=O)CC2)S1 51195,c1(C(=O)NC(CC=C)CNC(c2cnc(C)n2C(F)F)=O)cnc(CO)nc1C 51196,CCC(C)C(C(=O)NCC1COCCN1C)NC(C1OCCC1C(C)C)=O 51197,N1(C(c2ccc(NCC)cc2)=O)CCCC(C)C1CNC(c1ccccc1)=O 51198,c1(-c2ccc(C(=O)NC(CNC(C3CCSC3)=O)CO)s2)cccc(F)c1 51199,C1(C(=O)NCC(CN(C(COCC(C)C)=O)C)C)CCC(N(C)C)CC1 51200,C1(NC(CCN(C(=O)C(c2ccn(C)n2)C)CC=C)=O)CCCC1C(C)C 51201,C1(CC(=O)NCC2(O)CN(C(Cc3cnn(C)n3)=O)C2)CC2C=CC1CC2 51202,C1(CC(=O)NC2CC(N(C(CSCC(C)C)=O)C)C2)CN(C)CC1O 51203,O=C1NC(=O)C2CN(c3ccncc3S(=O)(=O)NCCNC3CC3C3CC3)CC12 51204,C1(OCC)CC2CCC1C2.n1(CC(=O)OCC2CC2)cccn1 51205,CC(=O)N=c1nc(C2CCN(C(C3CCN(C(=O)C(C)C)CC3)=O)CC2)[nH]n1C 51206,N1(C(c2ccc(OC)cc2C)=O)CCN(C(=O)C=CC=C(Cl)Cl)C(C)C1C 51207,C(C)(CCC(=O)NCCCCCO)NC(C1ON=C(C)C1)=O 51208,N1(C(C2CC2F)=O)CCC2(CCN(S(=O)(=O)c3ccc(O)cc3)CC2)C1 51209,c1(NC(=O)NC(C2CCOCC2)C)ccc(C#N)c(Cl)c1 51210,Cc1cccn2cc(C(=O)NCC3CCN(C(C4CCO4)=O)CC3)nc12 51211,C1(C(N(CC(C)NC(=O)C(C)(C)N(C)C)CC)=O)CCC(O)CN1C 51212,Cc1ccc(C(C)C(=O)NCc2nc(CNC(=O)CC3C=CCC3)cs2)cc1 51213,C1(C(C)NC(c2ccc(C)o2)=O)CN(C(=O)CC23COCC(C2)C3)CCO1 51214,c12cc(ncn1)C(=O)N2CC1CCCC(C(=O)OC)C1.C1(C)(CCCO)CNC1 51215,C1(C(=O)NC(CC=CC)CO)CN(C(c2cc(C(F)F)[nH]n2)=O)C(C)(C)C1 51216,C1(NC(CC(C)C2CCCO2)=O)CCC(C)N(C(=O)Cc2cnn(C)n2)C1 51217,N1(C(C=C(CC)CC)=O)CCC(NC(C23CSCC2C3)=O)C1C1CC1 51218,O=C(C=C(Cl)Cl)NCC1CC1CNC(c1sccc1-n1cccc1)=O 51219,Cc1nccn2c(C(N3CCNC(=O)C3c3ccccc3Cl)=O)cnc12 51220,c1(C(=O)NC(CNC(C(CC=C)C)=O)CO)cccc2[nH]c(C)cc12 51221,c1(N(CC(CN(C)C)O)C)ccc(Br)c(S(=O)(=O)NC2CN(C)C3(CCC3)C2)n1 51222,c1(C2(NC(=O)NCc3cc(Cl)cs3)CC2)ccc(F)c(F)c1 51223,N1(C(C2CCN(CC)CC2)=O)CCCC(O)(Cc2nc(C3CC3)no2)C1 51224,N1(C(C(C=CC)O)=O)CCOC(CCCNC(C2(SC)CCC2)=O)C1 51225,C1(CC)COC(C)(C)CN1C(=O)C1=CCN(C(=O)CC2CCCCCC2)C1 51226,C1(CNC(COCCC)=O)CCCCC1NC(=O)Cc1ccc(Cl)s1 51227,C(=O)(C1=NOC2(CCC2)C1)N1CC(C)C(C(=O)NC2(c3nncn3C)CC2)CC1 51228,N1(C(CC(=C=C)C)=O)CC(C2CCCCN(C(C3CCc4n[nH]cc4C3)=O)C2)C1 51229,c1(CC)cc(C(N2CC(Cc3ccoc3)C2)=O)nn1C.C12(CC1)CC(=O)N2 51230,C1(C(N2CCC(SC)CC2)=O)CCN(C(=O)Cc2nc(C3CC3)n[nH]2)C1(C)C 51231,C(=O)(C1=CCOC1)N(C1CC(NC(C(C)Cn2cccn2)=O)C1)C 51232,c1(C2C(NC(C3NCCC3C(F)(F)F)=O)C2)ccc(Cl)cc1 51233,c1(C(C)C)cnc(C(=O)N(C)CCOCCNC(=O)C(O)C(C)C)nc1 51234,C1(NC(C(COC)C)=O)CCS(=O)(=O)C12CN(c1nc(C(C)C)ncc1Br)C2 51235,c1(C(=O)NC2(COC)CCCN(C(=O)CC(C)F)C2)ccc(C)c([N+](=O)[O-])c1 51236,C(CCC(C)(C)NC(=O)CNC(=O)C(C)CC)NC(CC(=C)I)=O 51237,c1(OCC(=O)N(C2CC(C(F)(F)F)C2)C)cccc(C(=O)NC)n1 51238,C1(NC(c2c(C)ccc(Cl)c2)=O)COC2(C1)CN(C(=O)C(c1ccccn1)C)C2 51239,Cc1cccc(Cn2cncn2)c1-n1nc(CCN(C)C)nc1CCCC(C)(C)C 51240,C1(NC(C2CC(ON(C(C)C)C)C2)=O)CCN(C(c2n[nH]cc2Cl)=O)C1 51241,c1(C(N2CC(C)C(NC(=O)Cc3cnn(C)c3)CC2)=O)ccn2nccc2n1 51242,C(C)(C)(CC(F)C(=O)N(C)CC1CCOC(C)(C)C1)NC(C(C(=O)OC)OC)=O 51243,CN1CCN(C(=O)CN2CCCC2=O)CC1C(=O)NOCc1ccncc1 51244,C1(C(N2CC(O)(CCNC(c3cnc(C4CC4)s3)=O)C2)=O)CC2(C1)CC2(F)F 51245,CCCC(C)(O)C(=O)NCC1CCC1NC(c1ccc(N)c(CC(C)C)c1)=O 51246,CC1CC(NC(=O)CC2CCN(C(C3CC(F)C3)=O)C2)C(=O)O1 51247,N1(C(CSCC(=O)OC)=O)CCC(NC(=O)CC2CC(N(C)C)C2)C(F)(F)C1 51248,CN1CCC(C)(C(=O)NCCOC2CCN(C(=O)CSCCC(F)(F)F)CC2)CC1 51249,C=CC(CC)CC(=O)NCC1CCN(C(c2cc(C(F)(F)F)ccc2O)=O)C1 51250,c1(OC)c(C(=O)NCCCCCNC(c2c(Cl)cnn2C)=O)ccnc1Cl 51251,Cc1ccnc(O)c1C(=O)N(CCNC(C12CCCCC1C2)=O)C1CC1 51252,Cc1c(C(N2CC(F)(C(=O)NC3(C)CCCC3(F)F)C2)=O)cccc1O 51253,C=CCCCC(C(=O)NCCCCC(F)(F)F)NC(C1CC2(CC2)CO1)=O 51254,[N-]=[N+]=NCCCCC(=O)NCC1(NC(=O)CC2CC2(Cl)Cl)CCOC1 51255,C(CCCCC(=O)NCCC1(O)CCN(C(=O)CCn2ccnc2)C1)NC(N)=O 51256,C1(C(=O)NC(C2CN(C(c3ncoc3-c3ccon3)=O)C2)C)C(C)(C)C1(C)C 51257,c1(OC)ccccc1C(CNC(C1CCC2CC12)=O)NC(C12CC(CO1)C2)=O 51258,C=CC1(CC(N2CCC(C)C2CO)=O)CN(C(c2nn(C)cc2C)=O)C1 51259,C(=O)(CC(C)CNC(=O)COC(C)=O)NC1(CC=C)CCOC1 51260,CCCS(=O)(=O)CC(=O)NCC(C)(O)CNC(C1CC2(CCC2)CO1)=O 51261,N1(C(c2c(C)nc(N)cn2)=O)CCC2(CCC(NC(=O)C#CC3CCOC3)C2)C1 51262,c1(CC)ccc(CC(=O)NCC2CC2NC(c2cc(=O)n(C)cn2)=O)cc1F 51263,C1(C(N2CC(CNC(c3ccc[nH]3)=O)C(F)(F)CC2)=O)CC2CCCCCCC12 51264,c1(C(N2CC(CNC(C(C=C)O)=O)OCC2)=O)ccc(C)c(S(=O)(=O)CCO)c1 51265,Cc1ccc2c(C(=O)N(C)CCN(C(=O)CC3CC(=O)C3)C)coc2c1 51266,N1(C(C(CC=C)CC)=O)CC2COCCC2(NC(c2cnc(Cl)s2)=O)C1 51267,c1(C(=O)NCCN(C(C2N(CC)CC2)=O)C2CC2)c(C2CC2)cccc1F 51268,N1(C(c2cc(CNC(=O)CCc3cncnc3)no2)=O)CCC(C2CCCC2)C1 51269,C(C(CC)CO)NC(C1(N(C(COCCC=C)=O)C)CC1)=O 51270,c1(C(N2CCC(OCC)C2)C(=O)NCC2CC2)sc(C)nc1C 51271,CCCCC(O)CC(=O)NCC1(Cc2ccc(F)c(O)c2)CCCN1C(=O)C1CC1 51272,c1(CCC(=O)NCC(O)CNC(C2(F)CCCC2)=O)ccc2c(c1)OCO2 51273,C1(C)(C(=O)NCC(CNC(C2(CC#C)CCCC2)=O)O)Cc2ccccc2N1 51274,C1(C(N2C(C)COC(C)C2)=O)CCCC2(CCCC2)O1 51275,CC1CN(C(c2nn(C(C)(C)C)cc2Cl)=O)CCN1C(C1CC(=O)NC1(C)C)=O 51276,c1(C(=O)OC)c(F)cc(Br)c(CS(C)(=O)=O)c1F 51277,c1(C(=O)NC2CC2NC(c2cnns2)=O)cc([N+](=O)[O-])c2nsnc2c1 51278,c1(OC)nccc(C(N2CC(OC)CC(NC(=O)CSS(C)(=O)=O)C2)=O)n1 51279,Cc1nn(C)cc1C(=O)NCCCC1CCCN1CC(O)COCc1cccs1 51280,c1(NC)cncc(C(N2CC3C(CNC(C4(C(C)(F)F)CC4)=O)C3C2)=O)c1 51281,c1(NC2CCC(=C)CC2)cc(Br)ccc1S(=O)(=O)NC1CCOCC1C1CC1 51282,Cc1cccc(CN2CCC(C)(CN)C2)c1Br 51283,N1(C(C=NOC)=O)CCCCC1CC(=O)NC1C(C)C1C 51284,C(C(CC(=O)NC(CC1CC1)CO)NC(=O)C(C)c1cc[nH]n1)OC 51285,C1(CNC(c2ccns2)=O)COC(CNC(c2ccc(-c3ccccc3)o2)=O)C1 51286,c1(C(N2CCN(C3CCN(C(C)C)C3=O)C(C)C2)=O)cc2cccnc2[nH]1 51287,CCC(COC)C(=O)NC1CN(C(c2ccc(-c3csnn3)cc2)=O)CC1C 51288,C(=O)(C(F)C(C)(C)O)NCC1C(C)CN(C(=O)C=CCN2CCCC2)C1 51289,C1(C(NOC(C=C)C)=O)N(C(c2csnn2)=O)CCCC1(C)C 51290,N1(C(=O)CCc2ccccc2)CCC(C2CCCN(C(c3ccco3)=O)C2)C1 51291,Cc1sc(C(F)(F)F)nc1C(=O)NC1CC1CNC(=O)C(C)CC1CCCC1 51292,c1(C(=O)NC2CC(CNC(C3(C)N(C)CC(O)C3)=O)C2)ccc2nc(=N)[nH]n2c1 51293,C1(NC(c2n(C)ncn2)=O)CC2CN(C(=O)Cc3c(Cl)cnn3C)CC12 51294,C#CC1CN(C(c2cc(F)n(C)n2)=O)CCN1C(C1CCN(C)C1=O)=O 51295,C1(C(=O)NCC(C)N(C(=O)CCC(C)(C)N(C)C)CC)CCc2cnnn2C1 51296,CCCCCCCCCCC(=O)N1CCCC(N(C(=O)C2=CSCS2)CCO)C1 51297,N1(C(Cc2c(C)nsc2)=O)CCC(NC(C2(c3ccc(F)cc3)CC2)=O)C(F)C1 51298,Cn1cc(CC(=O)NC(C)(C)C(=O)NCCC2(O)CCC2)nn1 51299,N1(C(CCOCC#C)=O)CC(CNC(c2c(NC(C)=O)c[nH]c2C)=O)CC1C 51300,c1(C(=O)NC(CC(=O)N2C(C)(C(=O)NC)CC2)COC)coc2c1COC2 51301,c1(C(=O)NC2CC(NC(C3(CCOC)CC3)=O)C(O)C2)ccc(F)cc1C(N)=O 51302,N1(C(C)(C)C)CCC(O)C(CN2CCCCC2C(=O)Nc2ncc(C#N)s2)C1 51303,C1(O)(CN(C(=O)CC2CN3CCC2C3)C)CCN(C(=O)CN2CC3CC3C2)C1 51304,N1(C(c2ccc(OC)cc2)=O)CC(C)C(C)(CNC(=O)CCCCSC)C1 51305,CCCC(O)C(=O)NCC1(CNC(=O)C(C)SC)CCOCC1 51306,CCC(C)(CCC(C)C)C(=O)N1CCOC(C(N2CCC(F)(F)C2)=O)C1 51307,c1(C(=O)NC2C(C#N)CN(C(c3ccno3)=O)C2)ccc2ccccc2n1 51308,CCC(CC(=O)NC(C(=O)NC(C)COC)c1cccs1)C(F)F 51309,C1(CNC(COc2cn(C)nc2)=O)CN(C(=O)CC2C(C)(C)C2(C)C)CC1(C)C 51310,N1(C(C(C)C2CCC2)=O)CCCC(C2CN(C(c3cccc(C4CC4)n3)=O)C2)C1 51311,N1(C(C2COCCN(C(c3c(CC)ncs3)=O)C2)=O)CCNc2ccccc21 51312,c1(C(N2CCC(NC(c3n(C)ccn3)=O)C(F)C2)=O)cncc2[nH]ccc12 51313,C1(NC(C)=O)CCN(C(C2CCN(C(C3CCCC3C)=O)CC2)=O)CC1 51314,C1(C(C)(C)C)CC(C(=O)N2CC(CNC(=O)CCc3cn[nH]c3)C(C)C2)=NO1 51315,c1(C(=O)NCC2(C(C)(C)C)CCN(C(c3c(C)ncs3)=O)C2)ccc(N)cc1Cl 51316,c1(C(N2CC=CC(NC(=O)C3=CCC3)C2)=O)ccc2c(=O)ccoc2c1 51317,C(=O)(C#CC1(C)CCCO1)NC1CC2CN(C(c3nn(CC)c(O)c3)=O)CC21 51318,c1(N(C2CCOCC2)C(N(C2CC2C2CC2)C)=O)ccc2nsnc2c1 51319,c1(C(N2CCC(CNCc3ccc(Cl)cc3)CC2)=O)cc(C(F)(F)F)ccc1O 51320,N1(C(C2(NC(C3CCN(CC)C3)=O)CCN(C)C2)=O)CCCN(C=O)CC1 51321,c1(CC)noc2ncc(C(N3CCN(C(C4CCCSC4)=O)C(C)C3)=O)cc12 51322,c1(C(=O)NC2CCN(C(C3OCCN(C)C3)=O)C2)ccc2c(n1)OCC(=O)N2 51323,S(=O)(=O)(C1CN(C(=O)NCC2CCOC2(C)C)CC1)NC 51324,C(=O)(C(C#N)C(C)C)N1CCC(C(C(=O)NC(c2nccn2C)CC)F)C1 51325,C(=O)(CCCCCNC(=O)C(C)C)OCC.C12CC1CNC(=O)CNC(=O)N2 51326,c1(NC(CC=CC)=O)cc(C(=O)OC)ccc1C 51327,N1(C(c2c(CC)nco2)=O)CCOC(CCNC(=O)C(C)CF)C1 51328,c1(OC)cccc(C(=O)NC(C2CCN(Cc3cnc(C)s3)CC2)C)c1O 51329,C1(C(=O)NC(C(C)NC(C(CC=C)(F)F)=O)CO)CN2CCN1CC2C 51330,Cc1nc(N(CCCO)C(C)C)ncc1-c1ccc(COCC(F)(F)F)cc1 51331,C=CC(CCC)CC(=O)N1CCOC(C)C1C(N1CCC(OCC)C1)=O 51332,S(=O)(=O)(c1ccc(OC2CCOCC2)cc1C)NCCc1c(C(N)=O)cccc1 51333,N1(C(c2c(C)nns2)=O)CCCN(C(c2nc(Cl)sc2Cl)=O)CC1C 51334,N1(C(c2cc(CC)[nH]n2)=O)CC(CNC(=O)C(N2CCOCC2)C)CC(C)C1 51335,c1(OC)cc(N)c(F)cc1C(=O)NCC1CCCN1C(=O)CCCN(C)C 51336,Cc1ccc(Cl)cc1CN1CC2CC2(C(=O)NC2CNC(=O)C2)C1 51337,C1(CC(=O)NCC=CCl)CCCCN1C(c1ccc(Cl)o1)=O 51338,C1(NC(CCc2c(C)cccn2)=O)CCN(C(C2(C)CCCC2)=O)CC1(C)C 51339,C(N=c1[nH]c(=N)[nH]c(=NC2CCN(CCF)C2)[nH]1)C1CC(CC)C1 51340,CC1C(NC(c2ccccc2)=O)C(C)CCN1C(c1cnc2cccnn12)=O 51341,C1(C(=O)OC)CC(CN)CN(C(=O)C(CC)(CC)OC)C1 51342,C=CC(C(=O)N(C1CC(C(=O)NCC2(C(F)(F)F)CCCC2)C1)C)OC 51343,C1(F)(CNC(C)CC2CCC2)CCN(C(=O)OC2CCN(c3ccccc3)C2)C1 51344,N1(C(CCCC2CCC(=O)N2)=O)CCN(Cc2cn(C(C)C(=O)O)nn2)C(C)C1 51345,C1(O)(CN(C)C(c2occc2Cl)=O)CCN(C(=O)CCC(N)=O)C1 51346,c1(NCC)cncc(C(=O)N(C)CCOCCNC(=O)CCc2cn(C)nn2)c1 51347,C(CN=c1[nH]c(=NC(C)C(c2ccco2)NCC)[nH]c2c1CCC2)SCCOC 51348,c1(NCC2(COC)CC2)nc(N2CCC3(CC(=O)NC3=O)C2)nc2scnc12 51349,N1(C(C(COC)Cl)=O)CC2(C(N3CCNC(C)(C)C3)=O)CC1CO2 51350,c1(C(N(CCCNC(=O)CC2CC3(CC3)C2)C)=O)sccc1C#N 51351,C1(F)(CNC(CCOCCOC)=O)CCN(C(c2cc(F)ncc2OC)=O)CC1 51352,C=Cn1nncc1C(=O)NC1CCC(NC(C2(CCC)CCC2)=O)C1 51353,c1(OC)cc(C)c(C(=O)NC2CN(C(=O)CCc3cnc(O)[nH]3)CC2O)c(C)c1 51354,n1(CC)nc(C)cc1C(N1CC(F)CC1C(N1CCC(O)(CC)C1)=O)=O 51355,C1(N(C(CCSCC)=O)C)CCCN(C(C)=O)C1.c12ccc(cn1)c(=O)[nH]2 51356,N1(C(C(C(C)NC(c2cc(=N)[nH][nH]2)=O)(C)C)=O)CC(O)C2(CCCC2)C1 51357,c1(C(=O)NC(C2CCN(C(C(C)=CC)=O)C2)C)cc(C)c(C)o1 51358,CCC(C)(C)C(C(=O)NCCn1cc(C(=O)NC2(CO)CCC(C)C2)nn1)OC 51359,N1(C(CC(C)P(C)(C)=O)=O)C(C)CC2CN(C(c3cccc4nc[nH]c34)=O)CC12 51360,Cc1sc(C(=O)NC2CC(O)CN(C(c3ccc(O)nc3)=O)C2)cc1S(N)(=O)=O 51361,C1(OC)CN(C)C(C)(C(=O)NCC(CO)NC(c2ccsc2SC)=O)C1 51362,N1(C(C(C)(F)F)=O)CCN(C(=O)CN2CC=CC2)CC(O)C1 51363,N1(C(c2cc(SC)oc2)=O)CCN(C(=O)CNS(=O)(=O)N(C)C)C(CC2CC2)C1 51364,C1(C(=O)OC)CC2CC2N1C(=O)C(N1CC2CC2C1)C 51365,CCC(C)(C)C(=O)C(=O)N(C(C)C)CC1CC1.C1C(=O)NOCCCO1 51366,c1(-c2ccc(C(=O)NCCN(C(=O)CCCc3ncco3)C)[nH]2)ccccc1F 51367,c1(C(N(CC(C)NC(=O)C(C)(O)c2ccccc2)CC)=O)ccc(C)nc1OC 51368,Cc1ccc(C)c(CN(C(c2cccc(Br)c2)C(=O)O)C)c1 51369,c1(C(=O)OC)cc(C#N)cnc1NC(=O)NCC(O)COc1cccc(Cl)c1 51370,c1(C(N2CC(C)(NC(C3CC(C#N)C3)=O)C2)=O)nnn2c1CSCC2 51371,c1(-c2cccc(COCC)c2)ccc(C(=O)NCC2CC2)c(C)n1 51372,Cn1ncc2c(N3CCC4(NC(=O)Cn5cnnc5)CCCC34)ncnc12 51373,C1(NC(=O)C(F)CC2CC2)CN(C(c2cccc(Br)c2)=O)CC2(CCC2)C1 51374,c1(C(=O)NC2CN(C(CC(CCC)O)=O)CC(C)C2)cc2ccc(F)cc2[nH]1 51375,C1(COC)(CNC(=O)C2=CCSC2)CCCN1C(c1ccc(C#N)s1)=O 51376,C[Si](C)(C)CC(C(=O)O)NCc1ccc2c(c1)COC2 51377,CCCC(CCCO)C(=O)N1CC(C)CN(C(c2cccs2)=O)CC1C 51378,CN1CCC(C(=O)NC2CCC(C(=O)NC3CC3=Cc3ccccc3)C2)CC1=O 51379,c1(C(N(CCN2C(=O)C(OCCC#C)O2)CC)=O)cnccn1.OC 51380,c1(C(N2CCCC(CCNC(CCCCCC)=O)CC2)=O)cc2cccnc2o1 51381,CCCCCC(O)CC(=O)N1CCCC(C2CCCCN2C(c2cnsc2)=O)C1 51382,CC(C)CC(O)C(=O)ONC(=O)CC1CCN1.CC(CO)C(C)C 51383,C1(NC(=O)NC2CCN(OC)CC2)CC(N=c2[nH]c3ccc(N)cc3s2)C12CCC2 51384,c1(CNC(C2(C)CN(C)C(=O)C2)=O)ccc2c(c1)CN(C(=O)CS(C)(=O)=O)C2 51385,c1(C(=O)NC2C(NC(C(CC)C)=O)C2)c(OC)cc(OC)cc1OC 51386,C1(C(N2C(CN(C)C(c3cnc(Cl)cc3I)=O)COCC2)=O)CCC(C#N)CC1 51387,c1(C(=O)NC2C(CNC(c3c(COC)nn(C)c3)=O)C2)cc2occc2n1C 51388,N1(OS(CC23CC(C)(OC2)C3)(=O)=O)CCCN2CCCC12 51389,CC(C)CC(C)N(C(=O)CCN(C(=O)CC1OCCO1)C(C)C)C 51390,CCC(C)(CCNC(=O)Cc1ccn(CC)n1)NC(C1CC1C(C)C)=O 51391,C1(N(C(=O)C(C)Cc2ccco2)CC(C)C)CCN(C(C2CNC(=O)N2)=O)CC1 51392,C1(C(N2CC(OC)C(NC(C3CC3C3(C)COC3)=O)C2)=O)CCC(O)CN1C 51393,c1(C(=O)NCC2C(CNC(C3(C(C)C)CC3)=O)C2)cnc2[nH]ncc2c1 51394,N1(C(Cc2cc(=N)[nH]cc2)=O)CCCC(NC(c2cccc(CO)c2)=O)CC1 51395,S(=O)(=O)(c1cccc(C2OCCO2)c1)Nc1cc(F)cc(C)c1Br 51396,CCC(CC1CCCC1)C(=O)NCC(O)CNC(c1cc(C(=O)OC)ns1)=O 51397,c1(N2CC(C)(C)C(NC(=O)COc3ccsn3)C2)cc2nncn2cn1 51398,C#CCC(O)C(=O)N1CCOC(Cn2cc(-c3ccn(CC(F)(F)F)n3)nn2)C1 51399,N1(C(c2ncn(CC)c2)=O)CCC2(CC1)CN(C(=O)CC1CC1)CC2CO 51400,c1(CCNC(=O)NC(CSC)(C)CO)cc(C)ccc1Cl 51401,C=C1COc2c(C(=O)NC3CC(CO)N(C(C4(N(C)C)CCC4)=O)C3)cnn2C1 51402,Cc1nc(Cl)ccc1NC(C1CN(C)CCN1C(=O)C(C)c1ccsc1)=O 51403,c1(OCCCOC)ncccc1CNC(c1nnc(C2CCNCC2)s1)=O 51404,C1(C(=O)NC(COC)C(=O)N2CC(N3CCC3)C2)CCC2(CC2)C1 51405,Cc1ccccc1C=CC(=O)NC1C2CC3C(C2)C13 51406,c1(NCC(N2C(C)(CNC(C)=O)CC(F)(F)C2)=O)ccc(S(N)(=O)=O)cc1 51407,C1(C(N2C(C)CC2)=O)CC12CCN(C(=O)C(C)CC#N)CC2 51408,CN1C(=O)CCC1CNC(c1occc1CNC(c1csc(F)c1)=O)=O 51409,N1(C(c2cccc(OCCC)c2)=O)CCN(C(=O)CSC)C(c2ccnn2C)C1 51410,c1(C(N2CCCC(N(C(=O)C(F)=C3CCCC3)C)CC2)=O)ccc2cncn2c1 51411,C=CCC(F)(F)CNC(=O)CN(C)C(C1CCN1C(C)(C)C)=O 51412,C1(C(N(C(C)CC(=O)N(C)CCC2CCCO2)C)=O)C2CN(C)CC12 51413,c1(NC(C)=O)ccc(Cl)c(C(N2CCOCC2CNC(=O)CNS(N)(=O)=O)=O)c1 51414,c1(-c2ccc(CN3CC(C(=O)OC)C(C)CC3)s2)cccc(F)c1C#N 51415,C=C(C)CC(=O)NCC(=C)CCNC(c1cncn1-c1ccccc1)=O 51416,C(=O)(CC(C)CC(=O)N1CCC(C)(C)C1C(=O)NCCCc1cc(C)no1)OC 51417,c1(CC=C)ccccc1C(=O)NC(C)C=CC(=O)NCc1c(C)noc1C 51418,C1(NC(C=Cc2c(C)ccs2)=O)CN(C(=O)C(=C2CCCCC2)F)CC12CCC2 51419,C1(C)(NC(C=CC(CC)C)=O)CC(NC(C2CCC(C(F)(F)F)O2)C2CCC2)C1 51420,c1(C(N2CCC(NC(C3ON=C(C)C3)=O)C(O)C2)=O)cc2ccc(F)cc2s1 51421,c1(C(=O)NC2CC(CNC(C3CC(F)(F)C3)=O)C2)nccc(Br)c1O 51422,CC(F)(CNC(=O)CCc1ccsc1)CNC(c1sccc1C1CC1)=O 51423,CCCC(C(=O)NCCCN(CCC)C(C1CCN(C)C1C)=O)NC(N)=O 51424,C1(NC(c2nc(C#C)sc2)=O)CS(=O)(=O)CC1NC(=O)CN(CC)CC 51425,c1(C(N(C2CCCN(C(C(C)NC(C)=O)=O)C2)CCO)=O)ccc(F)c(C)c1N 51426,c1(OCc2onc(-c3cn(C)nc3-c3ccnn3C)n2)ccc(F)c(F)c1 51427,CC1CN(C(C2CCN2CC(F)(F)F)=O)CC1(C)CNC(=O)CCOCC(F)F 51428,Cc1cnc2c(C(=O)NC3CN(C(=O)CO)CC34CC4)cccn12 51429,C1(CC(=O)Nc2c(CC)ncs2)CCN(C(=O)CNC(N)=O)C1(C)C 51430,c1(C(=O)NC2C(C)N(C(=O)CCc3cncc(F)c3)CC2)nc(Cl)ccc1N 51431,N1(C(C2C(C)CCC2)=O)CCC(C(N2CCC(O)(c3ccccc3)C2)=O)CC1 51432,N1(C(c2cc(C)c(C)[nH]2)=O)CCN(C(=O)CCC(N)=O)CC1C 51433,c1(CC)cccc(OCC(N2CCC(C)(NC(=O)CCS(C)=O)C2)=O)c1 51434,N1(C(C2CN(C(C)=O)C2)=O)CC(C(=O)NCC(C)(F)C(C)C)C(F)(F)C1 51435,c1(C2C(C(=O)NCC3CC(NC(=O)C(F)=C4CCC4)C3)C2)ccc(F)cc1F 51436,C(c1ccccn1)=CC(=O)NCC(CO)NC(C(C)N(CC(F)(F)F)C)=O 51437,CC(c1cccs1)=CC=CC(=O)NCC1(C)CCCN1C(=O)CO 51438,N1(C(C(=O)NC(C)C)=O)CCC2CC12C(=O)NC(CO)C(N)=O 51439,C#CCC(CC(=O)NCC#CC1CC1)NC(=O)CN1CCC(C)C1 51440,C(C)(c1ccco1)=CC(=O)N(CCC)CCNC(=O)Cc1ccn(CC)n1 51441,C1(NC(c2ncccc2Br)c2n(CC=C)nnn2)CC2(C1)CC21CCC1 51442,c1(C(N2CC3C(CNC(C(C)OCC#C)=O)(C3)C2)=O)c(C)cc(C)cc1O 51443,C1(F)(C(N2CCC(OCC(C)C)C2)=O)CCCN(C(c2c[nH]nc2Cl)=O)C1 51444,c1(C(=O)NCCN(CC(C)O)C(=O)Cn2ncnn2)cc(F)cc(S(N)(=O)=O)c1 51445,c1(C(=O)NC2CN(C(c3cc(CC)[nH]n3)=O)C(C)C2)ccc(=O)n2c1COCC2 51446,C1(C(=O)NC(C23CCC(CC2)C3)CNC(COC(CC)C)=O)CCOC(=O)CC1 51447,c1(OCCN(C)C)ccc(C(N2CC(NC(=O)Cc3ccsn3)C(O)C2)=O)cc1N 51448,c1(C(=O)NC2CN(C(C3(F)CC=CCC3)=O)C2)cc(O)nc(O)n1 51449,C1(NC(C2C(C)(CC)C2)=O)CC2CCC(C1)N2C(C1(N(C)C)CC1)=O 51450,c1(C(=O)NCC(CC=C)NC(C2CCCC(O)C2)=O)cccc2c1CCCN2 51451,C1(C(=O)NC2CC(NC(C(C)OCC=C)=O)C2)CCC2(CC1)CC2(F)F 51452,Cc1cc(C(=O)NCCC(O)CNC(=O)CC(C)C)n(C2CC2)n1 51453,CCCC(C)(O)C(=O)NCCN(C(c1nc(C)nn1C)=O)Cc1ccc(Cl)nc1 51454,C1(NC(=O)NC(c2ccc(OC)nc2)C)(CO)CCCCC1C 51455,N1(C(C2C(C)CCO2)=O)CC=CC(C(=O)N(C)CC2CC2)C1 51456,CC1CN(C)CC(C(=O)NCC23CC(NC(C4CC(=O)N(C)C4)=O)(CCO2)C3)O1 51457,C(c1cccc(Br)c1)=CC(=O)NC(CC)CNC(=O)Cc1ncn(C)c1C 51458,C(CC(C)C)(C(=O)Nc1cncnc1C1CC1)ONC(C(C)NC(C)=O)=O 51459,c1(CNC(c2cccc(C)n2)CC)nn(C)c(Cl)c1I 51460,C(=O)(C(O)CC[S+](C)C)NCc1cn(CC(C)NC(c2cc[nH]n2)=O)nn1 51461,Cc1nnccc1C(N1CCC(N2CCN(C(c3cnn(C)c3C)=O)CC2)C1)=O 51462,c1(OC)cccc(C=CC(=O)NC2CC2NC(=O)CCc2nnc(S)nc2O)c1 51463,Cc1c(C(=O)NCCc2n[nH]cc2C(=O)NC2COCC2C)nnn1C 51464,C1(NC(c2c(OC)nccc2)=O)CC(F)CN(C(C2CCC(=O)NC2)=O)C1 51465,C1(NC(C2CCC(=C)CC2)=O)CCN(C(=O)Cn2cc(C(F)(F)F)nn2)C(C)C1 51466,C1(C(=O)NCC(C)C(=O)NC(c2ccncn2)C)C(C)(C)C1(F)F 51467,C1(F)(C(=O)NC2C(C(C)C)CCCC2)CCN(C(c2ccccc2)=O)CC1 51468,C1(CNC(=O)CSC(F)F)CN(C(C23CC4CC2C3C4O)=O)CCC1(F)F 51469,N1(C(c2cnc(CC)s2)=O)CC2(CC(CC(=O)N(CC)CC3CCC3)C2)C1 51470,c1(C(N2C(CNC(C=C(C)CCc3ccccc3)=O)CC2)=O)ccc(F)cc1O 51471,N1(C(c2cc(CC)ncn2)=O)CC2(C1)CN(C(=O)C(C)CCO)CC2CO 51472,CC1(CN2CCCC2)CCCN1C(C1CC=CCO1)=O.C12CCC(O1)CNC2=O 51473,N1(C(C=CC=CC)=O)CC2C(CNC(c3c[nH]c(C(=O)OC)c3)=O)C2C1 51474,C1(NC(C2N(C(C(CN(C)C)O)=O)CCN(C)C2)=O)CCCC(C2CC2)C1 51475,c1(C2C(C(C(=O)NCCC#N)N(C)CCC3CC3)C2)ccc(F)c(F)c1 51476,C(CCCC(=O)NC(C1CCCN1C(c1ccsc1COC)=O)C)OCC 51477,c1(C(N(C2CCN(C(CN(CCOC)C)=O)CC2C)C)=O)cc2cccnc2o1 51478,CC1C(NC(=O)CC2CCCCCC2)CCCN1C(c1cscn1)=O 51479,Cc1nnc2n1CC(C(N1CCN(C(C3CC(F)(CO)C3)=O)CC1CO)=O)C2 51480,N1(C(C(NOC)=O)=O)CCC(C=CC(=O)N(CCN=[N+]=[N-])C)CC1 51481,C1(NC(CCN2CCC(C)CC2)=O)CCCN(C(C2CCO2)=O)CCC1 51482,C1(N(C(=O)C(C)(C)NC(=O)C(F)(F)F)C)CCCCN(C(C2(SC)CCC2)=O)C1 51483,CC(C)(CC(F)(F)F)C(=O)NCC1CN(C(c2cnn(C3CCC3)c2)=O)C2CC12 51484,C1(O)(CN(C)C(c2ccnn2CC#N)=O)CCN(C(=O)COC2CCOC2)C1 51485,C1(C)(CNC(C(C2CN(C(c3cn(C4CC4)cn3)=O)C2)OC)=O)CSCCO1 51486,CC1CN(C(=O)Cc2ccoc2)CC1NC(c1ccc(N2CCC(O)C2)cc1)=O 51487,c1(OC(C)C)c(F)cc(-c2ccccc2C(N2CC3CCC2C(O)C3)=O)cc1F 51488,C1(N(C(COCC(C)C)=O)C)CCN(C(=O)Cc2cncn2C2CC2)CC1 51489,N1(Cc2cn(C(CNC(c3cc(C(C)C)no3)=O)C)nn2)CCCNC1=O 51490,C(=O)(C(C)CC(C)C(C)=O)NC1C2OCC(NC(c3c(CC)n(C)nc3)=O)(C2)C1 51491,c1(CC)cncc(CNC(C2CC2CNC(C2CCCC(O)C2)=O)=O)c1 51492,C1(CNC(c2c(C)coc2)=O)CN(C(=O)C(O)C2CCCC2)CC1(F)F 51493,C(CO)(CCCCNC(c1ccnn1C(F)F)=O)NC(c1c(C(C)C)ncs1)=O 51494,N1(C(Cc2scc(C(=O)OCC)c2)=O)CCCC(C)(NC(=O)C(O)C(F)F)C1 51495,c1(OC(=O)NC(CC=CC)C(=O)NCC)nnc2n1CCC2.n12cc(nn1)CC2 51496,C1(NC(Cc2c(C)con2)=O)CC=C(C(=O)N2CC(C)C(C)C2C)C1 51497,N1(C(CCC#CC)=O)CCC2(CC(NC(=O)Cc3nc([N+](=O)[O-])n[nH]3)CO2)C1 51498,c1(C(=O)NC(C2CCN(C(c3c(C(C)C)csc3)=O)C2)C)n[nH]cc1[N+](=O)[O-] 51499,Cc1cc(Cl)cc(C(N2CC(NC(=O)CSc3ccncc3)CC(C)C2)=O)c1N 51500,C(=O)(CP(=O)(C(C)C)C(C)C)NC1CCN(C(C(CC2CC2)OC)=O)CC1F 51501,c1(OC)cccn2ncc(C(=O)N(CCO)Cc3cc(F)ccc3Br)c12 51502,c1(C(=O)OC)cc(C(=O)NC2(C)CN(C(=O)CC3CC3C)C2)cc(C)c1 51503,C(=O)(C(C)S(N)(=O)=O)NCC1(O)CC(C(=O)NCCc2cc(C)no2)C1 51504,N1(C(C2(C)CCCN(S(=O)(=O)CCBr)C2)=O)C2CCCC1COC2 51505,CCCCCC(CC)C(=O)NC1CN(C(c2cc(C)cnc2N)=O)CC1C1CC1 51506,C1(C(=O)O)(COC)CCCN(C(c2ccc(OCC(F)F)nc2)=O)C1 51507,C1(C(N2CCC(CN(C(C=Cc3nc(C)sc3)=O)C)C2)=O)Cc2ccccc2O1 51508,c1(C(N(CC(=O)NC2CCC2NC(C2CC23CC3)=O)C)=O)ccccc1Cl 51509,c1(-n2cc(CN(C)C(c3cc(O)cs3)=O)nn2)cccc(Br)c1 51510,CN1CCC(CC(NOC(=O)CCCn2cc(N3CCC(O)CC3)nn2)=O)CC1 51511,CC(C)(CC(F)(F)F)C(=O)N1CCN(C(=O)CCCCC(N)=O)C(C(F)F)C1 51512,c1(NS(C)(=O)=O)ccc(F)c(F)c1.c12cncc(c1)C(=O)N(N(C)CCO)C2 51513,N1(C(C=C(C)c2ccco2)=O)CCCC1C1CCCCN1C(=O)Cc1ccco1 51514,c1(OC)cc(NC(C2CC(NCc3nccs3)C2)=O)[nH]n1 51515,c1(C(N2CCC(N(CCNC(C3C(C)C3)=O)C)C2)=O)cnc2n1CCCC2C 51516,C1(C(=O)NCCn2cc(CO)nn2)CC12CCN(C(=O)C=Cc1cscn1)C2 51517,Cc1cc(=NCCCN2CCCC2)[nH]c(N2CC3CSCC3(C)C2)n1 51518,N1(C(C(CC(=C)Cl)NC(=O)Cc2ccn(C)n2)=O)CC(=O)NC(C)(C)C1 51519,c1(C2C(C(=O)NCC(CNC(c3cc(OC)ns3)=O)(C)C)C2)cccc(C#N)c1 51520,C1(C(N2CC(OC)C(C(=O)NC3C(C)(C)C3(C)C)C2)=O)CCCCNC1=O 51521,c1(N(C)Cc2cccc(OC)c2OC)nccc(=NC2CCCC2S(C)(=O)=O)[nH]1 51522,C1(C)(CC(=O)NCCCCC=C)CCN(C(c2ncsc2C)=O)C1 51523,N1(C(CCCSC)=O)CCC2(C1)c1[nH]cnc1CCN2C(=O)CCc1nccs1 51524,N1(C(N2CSCC2CC2CCC2)=O)C(C(=O)NC(C)(C)C)CCC12CC2 51525,C1(C(N(C(C#C)C)C)=O)C2CCC(C2)C1NC(C1CCC1C#N)=O 51526,C=CCC(C(=O)NC1CC=C(C(=O)NC2COC(C)(C)C2)C1)C(C)C 51527,N1(C(C(C)n2cccn2)=O)CCC2(CC(C(=O)Nc3cncc(Br)n3)=NO2)C1 51528,c1(CC(C(=O)N(C2CCN(C(c3cnc(CC)[nH]3)=O)C2)C)C)c(C)n[nH]c1C 51529,N1(C(CC=CCNC(C(C(C)C)CN(C)C)=O)=O)CCC2(CC(F)C2)C1 51530,C1(CCC(=O)NCC(C2CCCC2)NC(C(C)N(C)C)=O)CCN(C)CC1 51531,C12(C(=O)NC(CCCC)CNC(=O)C(F)n3ccnc3)C3CC(CC13)C2(F)F 51532,N1(C(c2c(OC)cncc2)C(=O)NCC2CCOC2)CC(CO)C(C2CC2)C1 51533,c1(CC(OCC)OCC)cn(Cc2ccc(C(=O)N(C(C)C(F)F)C)o2)nn1 51534,C1(C(=O)NC(CC=C)CNC(=O)C=CCN2CCOCC2)CCC(C(=O)OC)CC1 51535,c1(C(N(C2C(NC(CC(CC)C3CCC3)=O)CCCC2)C)=O)ncnc(C)c1C 51536,C(CC(C)(C)NC(=O)CNC=O)NC(CN(c1ccccc1)C)=O 51537,C1(NC(C)=O)CCCCN(C(c2cc(C)n(C3CC3)c2C)=O)C1 51538,N1(C(c2c(C)nn(C)c2)=O)CCc2c(C(N3CCCCC(O)C3)=O)csc2C1 51539,CCCCCC(O)CC(=O)N1CC2CCCC2(C(=O)NCC(C)C(C)(F)F)C1 51540,c1(C(=O)NC2C(C)N(C(=O)CCc3ccc(Cl)nc3)CC2)ccc2c(c1)COC2 51541,c1(OC)cncc(C(N2CCOC(CNC(C3CC(=O)N(O)C3)=O)C2)=O)n1 51542,Cc1ccc([N+](=O)[O-])cc1C(=O)NCC1(CNC(=O)C(CO)C(F)(F)F)CC1 51543,C(CNC(=O)C(C1CCCCCC1)C)(CC(C)C)NC(CC1(C=C)CCC1)=O 51544,C1(C(=O)NCC(COC)O)CCCN(Cc2ccc(CN(C)C)cc2)C1 51545,C12(C(N(CCN(C(=O)CCc3ccnn3C)CC)CC)=O)CC(CO1)C2(C)C 51546,c1(C(C)N(C(c2cnc(N(C)C)nc2)C(=O)NCCN(C)C)C)ncc(Cl)n1C 51547,c1(CCCC)nc(C(=O)NC(C)(C)CNC(=O)CCc2nc(CC)no2)cs1 51548,c1(CC(=O)NC(CCNC(CC(CC)SC)=O)C)ncn2c1CCCC2 51549,CC1CCC(C(=O)NCCn2ccc(C(=O)NCC(F)(F)C(N)=O)c2)CC1 51550,c1(C(=O)NCCN(C(Cc2c(C)ccs2)=O)C)ccc2[nH]ccc(=O)c2c1 51551,C1(C(=O)NC(CN(C(C2(COC)CCCO2)=O)C)(C)C)CC2CCC(C1)C2 51552,C1(C)(COCC)NC(=O)N(CC2(C)CN(Cc3sccc3OC)C2)C1=O 51553,c1(CNC(C2(SC)CCC2)=O)c(C)nn2c1CN(C(=O)C(C)NC(C)=O)CC2 51554,Nc1cccc(C(=O)NCCCCCNC(=O)CCn2cccnc2=O)c1 51555,c1(CSCC(=O)NC(CC)CN(C(=O)CCOCC2CC2)CC)ccccc1 51556,Nc1ccc(F)c(C(N2CCC(NC(=O)Cn3cc([N+](=O)[O-])cn3)C(F)C2)=O)c1 51557,C(CC(C)C)(C(C(=O)NCC(F)F)N1CCSCC(C)C1)OC 51558,c1(CN(C)C(C2COCCN2C(=O)CC2CC2)=O)ccc([N+](=O)[O-])cc1 51559,c1(OC)cc(C)c(CNC(N2CCC(C)C3(CCC3)C2)=O)c(C)c1C 51560,n1(CC(=O)OCC)nc(C)c(S(=O)(=O)N2CC(O)CC2C(=O)OC)c1C 51561,c1(C(=O)NCC(F)CNC(C2(C(F)F)CC2)=O)cccc2ccnn12 51562,c1(C(=O)NCC2C(C)CN(C(C3CC(O)C3)=O)CC2)nc(Cl)c(=O)[nH]c1N 51563,C1(C(N(C(CCNC(Cn2ccc(C)n2)=O)C)C)=O)CC(=O)N(C2CC2)C1 51564,c1(C(=O)NC(CN(C(c2cnc(OCC)nc2)=O)C)CC)ccc(F)cc1C 51565,c1(C(N2CCCC(NC(c3cncc(F)c3Cl)=O)C2)=O)nc2cc(O)ccc2[nH]1 51566,N1(C(CCCCC#C)=O)CCS(=O)(=O)C(CCNC(=O)C(O)P(C)(C)=O)C1 51567,N1(C(C2C(OC)CC2)=O)CCC(NC(=O)CNC(c2cccc(C)c2)=O)C(C)C1 51568,C1(O)(C(=O)NC23CN(C(C=Cc4ccc(C)o4)=O)C(CC2)C3)CCCC(C)(C)C1 51569,c1(C(=O)OC)ccnc(C(N2CCNCC2C)C)c1F 51570,S(=O)(=O)(c1cc(Br)c(Br)s1)N1CC2(CCN(Cc3cncc([N+](=O)[O-])c3)C2)C1 51571,C(=O)(C(CC1CC1)NC(=O)C(C)NC(=O)CCc1cnco1)OCC 51572,C1(N2C(=O)C34CC(C3)(C4)C2=O)CCCC12CCNCC2.N#CC1(CO)CCC1 51573,c1(C(N(CC(O)CNC(C2(n3cccn3)CCC2)=O)C)=O)csc(Cl)c1 51574,C(C(=O)N=c1cc(C(N)=O)n(C)[nH]1)C1N(C(C(C=C)O)=O)CC(O)C1 51575,C(C(CNC(c1ccc(SC)cc1)=O)C(F)(F)F)NC(CCCC#C)=O 51576,c1(C(N(C)CC2N(C(CC(C=C)C)=O)CCCC2)=O)cc(C)cc2cccnc12 51577,C1(NC(c2n(C)ccc2)=O)C=CCCC1C(N1CCC2CCC12)=O 51578,c1(OCC(=O)N(C(CN(C(c2c(C)c[nH]n2)=O)C)C)C)ccccc1C(C)(C)C 51579,c1(NC(c2ccc(CNC(C(CC)n3cncn3)=O)o2)=O)ccc2c(c1)COC2 51580,C(Cc1ccccc1)(CCCO)CN(C=O)Cc1n(CC)nnc1 51581,c1(COC)ncc(C(=O)N(CCCOCCNC(C2(CCF)CCC2)=O)C)s1 51582,c1(C(=O)NC2CCN(C(C3(C)CC(C)(C)C3)=O)CC2)ccc(F)c(S(C)(=O)=O)c1 51583,N1(C(C(c2ccc(C)cc2)CC)=O)CC2(CCC(CNC(=O)CC(C)F)O2)C1 51584,N1(C(CC(C)(C)C2CC2)=O)CCN2CCN(C(=O)C#CC34CC5C(C3)C45)CC2C1 51585,N1(C(C(C=C)(C)CC)=O)CCC(CNC(=O)C(F)CCCCC)C(C)(C)C1 51586,c1(N2CCCC(OC)CC2)nc2c(cc1C#N)CCOC2 51587,CCS(=O)(=O)CCN(C(c1cccc(Oc2ccc(F)cc2)c1)C(=O)NC1CC1)C 51588,C1(NC(=O)OC(C)(C)C)CN(C(=O)CC(F)F)CC1C(=O)NC1CCCC1 51589,C(=O)(CCCCCNC(c1ccc(CF)cc1)=O)NCC(CC)OC 51590,C(C(O)CN(C(=O)COCCF)C)NC(C=CC)=O 51591,N1(C(c2c(CNC(C(CCCC)=O)=O)occ2)=O)CC(C)OC2(CCC2)C1 51592,C#Cc1ccc(C(N2CCC(CCNC(c3cnc(C)s3)=O)CC2C)=O)c(F)c1 51593,CCC(C(=O)N1CC=CC1CNC(c1ncccn1)=O)NC(N)=O 51594,c1(C(=O)NC2C(NC(C(CC)n3cccn3)=O)C2)cc(OC)c(Cl)cc1OC 51595,c1(C(N2CC(CCNC(Cc3n(C)ccc3)=O)OCC2)=O)cnc2[nH]ccc2n1 51596,Cc1c(C(=O)NC2CN(C(=O)CC3CCCOC3)CC2O)oc2c(Cl)cccc12 51597,C1(NC(C2(C(N)=O)CC2)=O)CCCC(NC(=O)C(c2ccc(O)cc2)=O)C1 51598,N1(C(C(C)OCC)=O)CCC(F)(CNC(c2ccc(N)cc2Br)=O)CC1 51599,c1(C(N(C2(C(=O)N(C(c3ccns3)C)C3CC3)CC2)C)=O)nc[nH]n1 51600,Cc1c(C(N2CCC(C(=O)NOC)C2)=O)cc(F)cc1Br 51601,c1(CN(C(C)C)C(c2ccc(-c3cc(O)n[nH]3)cc2)=O)nc(O)c2ccccc2n1 51602,C1(C(=O)NC(c2ncc[nH]2)(C)C)CN(C(=O)CN2CCC(=O)CC2)CC1(F)F 51603,N1(C(C2N(CC#C)CCC2)=O)CCCC2(CC(NC(C3CC(F)(CO)C3)=O)C2)C1 51604,N1(C(C(CO)NC(c2ccc(F)cn2)=O)=O)CC2CC1CO2 51605,C(CN=c1[nH]c(=NC2C=CCCCC2)[nH]c2c1COC2)N1CCC(OCCF)C1 51606,c1(CCC)c(C(=O)NCC(CC)NC(=O)CC2CC=CCN2C)cnn1C 51607,C1(N(C(C=C(CCC)C)=O)C)CC2CC1N(C(=O)CC(CC)C1CCC1)C2 51608,c1(C(=O)NC2CC(NC(C3CC3c3nc[nH]n3)=O)C2)ccc2c(c1)COCCN2 51609,C1(C2(O)CN(C(c3n[nH]cc3Br)=O)C2)(CNC(=O)C(F)=CCCF)CC1 51610,C(=O)(CCCC(F)F)N1CCC(NC(C(C(C)C)C)=O)CC1 51611,C1(OC)CCCC(C(N2CCCC2CCCNC(=O)Cc2c(Cl)cnn2C)=O)C1 51612,N1(C(CCC(C)N(C)C)=O)CC(C)N(C(C2CCCN2C)=O)C(C)C1 51613,C=CC(C)(CCOC)C(=O)N1CC2CC1C2CNC(C1(C(F)(F)F)CC1)=O 51614,c1(CC)ccccc1C(=O)NC1CCOC(C(=O)NOCCCN(C)C)C1 51615,c1(CNC(C2CC(=O)N(C3CCNCC3)C2)=O)ccnc(-c2ccccc2)c1O 51616,C(N=c1[nH]c(=N)[nH]c(=NCc2ccccn2)[nH]1)C1(N(C)C)CCCC1 51617,C1(C(C)=O)CC1(Cl)C(=O)NC1CC1NC(=O)COc1cn[nH]c1 51618,CCC(C)CC(C)C(=O)N1CCC(CC(N2CC(O)C(N=[N+]=[N-])C2)=O)CC1 51619,c1(OC)ccc(C(=O)NC2CC3CC(NC(=O)C=CC(F)(F)F)C3C2)c(C)c1 51620,N1(C(CCOCCOCC)=O)CCN(C(C2CCCC2)=O)CC2CCCCC12 51621,N1(C(CCc2ncc(C)[nH]2)=O)CCCCC(CNC(C2CCCN2C(C)C)=O)C1 51622,C1(NC(C(CC#C)NC(=O)C(C)CC2CC2)=O)CCCOC12CCC2 51623,N1(C(CCOCCC)=O)CCN(C(c2cn(C3CC3)cn2)=O)CCC1C 51624,C(C)(CC(C)C(F)F)NC(C(C)N(C(c1cc(CC)[nH]n1)=O)C)=O 51625,C1(O)(CC)CCN(C(C2(NC(=O)C(C(C)C)C3CC3)CCOCC2)=O)C1 51626,CC1=C(C(=O)N2CC(NC(=O)COc3ccccc3N(C)C)CC(C)C2)CCO1 51627,Cc1ccc2cc(C(=O)NC3CN(C(=O)COCCCF)C(C)(C)C3)[nH]c2c1 51628,C1(N(C(=O)CCC2CCCC2)CC)CCCC1C(=O)NCC1C(OCC)CC1 51629,N1(C(Cc2n(C)cnn2)=O)CCC2CN(C(C3CC(C4CC4)=NO3)=O)C2C1 51630,C(C(C)(C)C#CC(=O)N(C)CCF)NC(C(CC)N(CC)CC)=O 51631,C1(C)(CC)CCN(C(C2N(C(c3cnnn3C)=O)CCC2(C)C)=O)CC1 51632,C1(C(=O)NCC2(C)CC3CC3C2)CN(C(c2csc(F)c2)=O)CC1(F)F 51633,N1(C(CCc2n(C)ccn2)=O)CC2(CC(CNC(=O)Cc3cccs3)C2)C1 51634,c1(C(N(CC(CNC(CCCC(C)O)=O)C)C)=O)ccc(F)c(C#N)c1 51635,c1(C(N(C(C)C(=O)NC(C)C(C2CCCCC2)O)CCC)=O)ccc(=NC)[nH]c1 51636,C1(C(=O)NC(CC)CCOC)CC(NC(=O)Cc2csnn2)CCO1 51637,N1(C(C2(C)CC(C)C2)=O)CCC2(CC(NC(c3cccc4nsnc34)=O)C2)C1 51638,N1(CC(=O)NC2C=CCN(C(C(c3cccnc3)C)=O)C2)CCCCS1(=O)=O 51639,N1(C(C(C)SC)=O)CCC(C2CCCN(C(c3c(Cl)nn(C)c3Cl)=O)C2)C1 51640,C1(C)(C(=O)NCC2CN(C(c3sc(CC)c(C)c3)=O)CC2C)CCC(C)CC1 51641,C12(OC)CC3CC(C1)C(NC(=O)NCC1COC(C)C1)C(C3)C2 51642,N1(C(CSC2C(=O)OCC2)=O)CCC(NC(=O)Cn2cncn2)CC1 51643,CC(C)S(=O)(=O)C(C)C(=O)NCC1(O)CCCN(C(=O)C(F)(F)C2CC2)CC1 51644,N1(C(C(C)OC)=O)CCN(CC2CCCCN2C(c2ccnnc2)=O)CC1 51645,c1(C(N2C(C)CC(NC(CC(C)(C)SC)=O)C2)=O)cccc2[nH]cc(Cl)c12 51646,C(=O)(CC(O)C(C)C)N(CCCCC1(NC(C)=O)CC1)C(C=CCCC)=O.C(C)=C 51647,CON1CC(C(=O)NCC2CCCC2C(=O)NC2(C)CC=CC2)CC1=O 51648,C(CCCl)(CCCl)(c1n(CCOC)nnn1)NCC1(c2ccccc2)CC1 51649,c1(N(CCNC(c2csc(C(F)(F)F)c2)=O)CC)nc(O)c2ccc(Cl)cc2n1 51650,N1(C(C(C)(C2CC2)OC)=O)CC2CC(NC(c3cccs3)=O)CC1C2 51651,c1(NC(C(CCOC)C)=O)ccc(NC(=O)C(C)(C)n2ccc(C)n2)cc1C 51652,N1(C(CC(CC)OC)=O)CC(N(C(=O)CCOC)CC)C2(CC2)C1 51653,c1(C(N2C(C(=O)NCc3c(F)ccc(C)c3)CSCC2)=O)cc(C)c(C)cc1I 51654,O=C(CCCc1ccc2c(c1)OCO2)NNC(=S)NC1CCS(=O)(=O)C1 51655,C1(C(=O)NCC2CC(NC(=O)COc3cccnc3)C2)CCCC(=O)O1 51656,Cc1cc(N(CC(C)C(C)C)C)nc(=NCCc2ccc(C(F)F)cc2)[nH]1 51657,C1(CC(=O)N(C(CSC)C)C)(NC(C2CCCO2)=O)CCC1 51658,c1(CN2C(C)(COC)CCC2)cc(-c2cc(F)cc(F)c2OC)c(OC)c(Cl)c1 51659,C(CC(C(C)(C)C)NC(C1CCC(=O)C1)=O)N(C(c1cn(CCOC)nn1)=O)C 51660,N#CC1(C(N2CCCC(F)(C(=O)NCC#CCCO)C2)=O)CC(F)(F)C1 51661,c1(C(=O)NC(C)CC(C)NC(C2CCCC2c2ccccc2)=O)ccc(O)nc1 51662,C1(C(=O)NC(CNC(c2c(C)nc(C)[nH]2)=O)(C)C(C)C)CC2COCC2C1 51663,C(CC(C)CC)(C(=O)NCC(C)(C)C(F)(F)F)NC(c1c(CC)[nH]cc1)=O 51664,Cc1ccc(C(=O)NC2CC3C(NC(=O)CCc4ccc(C5CC5C)o4)C3C2)cn1 51665,C1(CN(C(=O)C(N2CC(F)(CO)C2)=O)C)CCCCC1O 51666,C1(C(=O)NC(C)C(=O)NCc2ccccc2)CCCN1C(C1CC(F)(F)C1)=O 51667,c1(C(C)C)c(Cl)nc[nH]c1=NCC1C(C)CCCN1C(=O)C=CCN(C)C 51668,N1(C(CCCOCC)=O)CCN(C(c2cc(OC)ns2)=O)CC1C1CC1 51669,N1(C(C(C=C)(C)C)=O)CCC2(CC1)CC(NC(=O)C(CC)n1nccc1C)CO2 51670,N1(C(C=CCOCCOC)=O)CC(C)N(C(c2cnc(C)s2)=O)CC1C.C1CO1 51671,c1(CN2CCCC(CC(=O)N(CCCCC=C)C)C2)cc(O)cc(Br)c1 51672,Cc1cccc(CC(=O)NC23CC2CN(C(C2(C(C)C)CC2)=O)C3)c1Cl 51673,N1(CC(Cc2ccccc2)OC)CCC(S(=O)(=O)N(C)C)C1 51674,N1(C(CCC(=O)NC)=O)CC(CO)C2(C1)CN(C(c1n[nH]cc1Cl)=O)C2 51675,c1(C(=O)NC2CC2)cc2n(n1)CCCN(C(c1ccc3nc(O)oc3c1)=O)C2 51676,c1(CC(N2C(CC)C(NC(=O)CC#N)CCC2)=O)c[nH]c2cc(C)ccc12 51677,C12(CNC(C(C)OCC#C)=O)CCCC1N(C(C1CC3(CCC3)C1)=O)CC2 51678,N1(C(c2cccc(Cl)c2F)=O)CCOC2(C1)CN(C(C13COCC1C3(F)F)=O)C2 51679,N1(C(C2(C=C)CC2)=O)CCC(NC(c2sc(SC)cc2C)=O)C(F)C1 51680,C12(C(=O)NC3(C(=O)NC(C(C4CC4)OC)C)CC3)CC(C#N)(C1)C2 51681,N1(C(C(C=C)(C)O)=O)CCCC(C)(C(=O)NC2CCOC2=O)C1 51682,CCC(C(=O)NCC(C)N(C)C(C1(C#N)CC1(C)C)=O)C(C)C 51683,c1(CNc2ccnc(SC)n2)cc(O)cc(O)c1.C12CCNCC1C2 51684,c1(C(=O)NC2C(CNC(c3c(C)ncn3C)=O)C2)cc(Br)cc2c1OCC2 51685,N1(C(CCCCC=C)=O)CCC2CN(C(=O)C(C)C(C)C)CCC12 51686,Cc1ccc(NC(C2CCCCN2C(=O)CC2CCCC(=O)C2)=O)c(C)c1 51687,c1(C(=O)NC(CCNC(c2c(C)snc2)=O)C)nn(-c2ccccc2)cc1Br 51688,c1(C(N2CCC(CN(C)Cc3nc[nH]n3)C2)=O)ccc(NC(N)=O)cc1 51689,C1(CNC(C(CC(C)C)O)=O)CN(C(c2ccccc2O)=O)CCC12CCC2 51690,c1(SC)ccc(C=CC(=O)NC(C2CCN(C(C3CCCCC3O)=O)C2)(C)C)s1 51691,C1(C(=O)NC2(C=C)CCC2)CCN(C(c2ncsc2NC)=O)C1(C)C 51692,c1(C(C)C)ccc(C(=O)NCC(=C2CN(C(=O)C(C#N)=CC3CC3)C2)F)c(F)c1 51693,Cc1ccc(Cl)c(C(=O)NCC2CC2CNC(C2(n3ccnn3)CC2)=O)c1O 51694,CC(O)C(C)(C)C(=O)N(CCC(C(C)(C)C)NC(=O)CN(C)C1CC1)C 51695,c1(C(=O)NCC2CC(OC)CN2C(=O)COCC(F)(F)F)c(F)ccc(F)c1Cl 51696,C12(CNC(C3(C(=O)NC4CC4)CC3)=O)CCC(C1)N(C(=O)C(C)n1cccc1)C2 51697,C1(CC)(CC)CC(C(=O)NCC2(C(N3CC(c4ncnn4C)C3)=O)CCCO2)C1 51698,c1(C(=O)NC(c2cn(C)nn2)C(=O)NCC(CC)N(C)C)cncc(C)n1 51699,Cc1cc(C(=O)NCC(CNC(=O)C(C)C(F)F)CO)c(Br)s1 51700,S(=O)(=O)(c1cccnc1N1CCn2cnnc2C1)N(CC(C)(C)N(C)C)C 51701,C(=O)(C1CCOc2ccccc21)N1CC(NC(=O)Cn2cccn2)CC(OC)C1 51702,C=C1CC2CCCC(C1)N2C(C1CCCN(C(c2csc(=N)[nH]2)=O)C1)=O 51703,C(=O)(C#CC1(C)CCCO1)NCC=C(C)C.c1(C(N2CC(CO)C2)=O)cc(Cl)n(C)n1 51704,c1(Sc2n(C(C)C)c(S)nn2)c(Br)ccc2c1OCCO2 51705,CCCCC(O)C(=O)N1CC(CN(C)Cc2ccc(C(C)=O)s2)C2(CC2)C1 51706,C1(C(=O)NC2(CF)CCN(C(C3CCC(C)(C)C3)=O)C2)CC2(CC(=O)N2)C1 51707,N1(C(c2ncc(CC)cn2)=O)CCC2CCCC12C(N1CC2C(C1)C2(F)F)=O 51708,c1(C(=O)NC(C2CCCCN2C(=O)CC2CSC2)C)ccc(S(=O)(=O)NC)cn1 51709,C1(C2CC2)(NC(c2cc(CNC(C3CC(CF)C3)=O)[nH]n2)=O)CCCC1 51710,C(=O)(C1CC(=O)Nc2ncn(C)c21)NC1C(C)N(C(=O)C=Cc2ccsc2)CC1 51711,Cc1nn(C)c(F)c1C(N1CCC(CNC(c2ccnc(OC(F)F)c2)=O)C1)=O 51712,CCC(CC(=O)N1CC(C)(C)CC1CC(=O)N(C)Cc1cnnn1C)CC(C)C 51713,CC(CC(=O)NCCCOc1ccccc1)N(C1CCCC1)C 51714,C(CC(C)C)(C(=O)NCC1CN(C(=O)COc2cccc(C(C)C)c2)C1)OC 51715,CCCCS(=O)(=O)N1CCC(C(=O)Nc2ncccc2C(=O)OC(C)C)CC1 51716,C(=O)(C#CC1(CC)CC1)N(CCNC(c1ccncc1N(C)C)=O)CC 51717,CC1CN(C(=O)Cn2ccnn2)CCN1C(=O)CC1(N(C)C)CCOCC1 51718,N1(C(c2ccn(C)n2)=O)CCC(C)(C(=O)Nc2cc(Br)ccc2O)CC1 51719,c1(C(N2CCC(NC(c3cc(C(C)C)no3)=O)C(O)C2)=O)ccc2snnc2c1 51720,N1(C(C(CCC)N(C)C)=O)CC(N(C(=O)C=Cc2cccnc2)C)C2(CC2)C1 51721,CC1(C)CC(C(N2CCC(C(C)(C)O)CC2)=O)CN(C(C2C3CCCCC23)=O)C1 51722,C12(C(N3CC(CC(C)NC(c4c(C)occ4)=O)C3)=O)COCC(C1)C2 51723,C(C(CC(C)C)C(=O)N1CCC(C)(C)C1C)NC(COCCC#C)=O 51724,CCC(CCC(=O)N(C)CC1(CO)CC1)NC(=O)CC1(C)CCCCC1 51725,C(=O)(C(C)CC(F)(F)F)NCCN(C(C(CSC)(C)C)=O)C1CC1 51726,C12(NC(CCc3onc(CCC)n3)=O)CCC(CC1NC(c1oncc1C)=O)C2 51727,NS(=O)(=O)c1cc(NC(=O)NC2C3CCCCCC23)c(F)c(Br)c1 51728,c1(C(=O)NCCCOCCC(=O)NC2CCC(N(C)C)C2)cnc(NC)cn1 51729,c1(NC(C2CCC(SC3(C(=O)OC)CC(O)C3)C2)=O)cnnc(OC)c1 51730,N1(C(CCSCCC)=O)CCN(C2CCCN(C(=O)C(C)NC(N)=O)C2)C(=O)C1 51731,c1(OC)cc(C(=O)NCC(C)CNC(=O)C(=O)NCCC(N)=O)ncn1 51732,c1(C(=O)NCC23CC(NC(C=C(C)C(F)F)=O)(C2)C3)c[nH]c2ncc(Br)cc12 51733,C(c1ncc(C)[nH]1)=CC(N1C(CN(C(C2CCC2(OC)OC)=O)CC)CCC1)=O 51734,Cc1cc(=O)c(C(=O)NCc2ncsn2)nn1-c1cccc(Cl)c1 51735,C1(NC(C2N(CC)CC2)=O)CN(C(C2CC(CC)=NO2)=O)CC1C 51736,C(C)(C)(C(=O)NCC1(CNC(=O)Cc2ccnn2C(C)C)CC1)OCC 51737,CCCCC(C(=O)N1CCN(C(=O)CSC)CC1c1ccccc1)NC(N)=O 51738,c1(CNC(c2occ(C)n2)=O)cnn2cccc(C)c12.C12CCCC1NC2=O 51739,N1(C(C2=C(C)CC2)=O)C(CC(N2CC3CCCCC23)=O)C2CCCC12 51740,c1([SH](C)CO)nc(C)ncc1-c1nc(CC(c2ccc(F)cc2)(C)C)no1 51741,c1(CC(=O)NCCC2CC(NC(CCc3ccc(C)s3)=O)C2)cn(C)nc1C 51742,c1(CC)csc(C(C(=O)NCCSn2cc(CN3CCOC3=O)nn2)OC)n1 51743,N1(c2n(CC)c(C3(Cc4ccccc4)CC3)nn2)CCN(C)C2(CCOC2)C1 51744,C=CCC(Cc1ccccc1)C(=O)NC1CCCC1NC(=O)CC(F)F 51745,c1(C(=O)NCC2(C)CCCN2C(C2CC2c2cncs2)=O)ccc(S(C)(=O)=O)o1 51746,N1(C(C(C)OCCOC)=O)CCN(C(c2ccon2)=O)C(C(F)F)C1 51747,c1(C(N2CC3C(CNC(C4(C)CCN(C)C4)=O)(C3)C2)=O)cc(F)ccc1C1CC1 51748,S(=O)(=O)(c1ccc(F)cc1O)NC(c1cnn(C)c1C1CC1)=O 51749,C1(NC(c2cc(F)n[nH]2)=O)CC(NC(C2CC(CF)C2)=O)C12CCC2 51750,C(C(=O)N(CCCCNC(=O)C(C)Sc1ccccc1)C)(C(C)C)NC(C)=O 51751,CC1C(=O)N(CC(=O)NC2(CNC(=O)Cc3nncs3)CCC2)C(=O)C1C 51752,C#CCCCCC(=O)N(C1CCC(NC(=O)Cc2ccnnc2O)CC1)CC 51753,N1(CC)CC(C(=O)NC2CCCN(C(C34COC(CCO3)C4)=O)CC2)CCC1=O 51754,n1(CC(=O)NC(C)CC(C)NC(C2CCC(=O)C2)=O)ncccc1=O 51755,C(C(C)(C)C(F)F)NC(C(C1CCN(C(=O)C=Cc2ccccc2)C1)C)=O 51756,c1(OC)cc(C(=O)NCC2CCN(C(c3coc(Cl)c3)=O)CC2C)cc(N)c1N 51757,c1(C(N2C(C(=O)NCC(C)(C)CCO)C(C)(C)CC2)=O)cccc2[nH]ncc12 51758,N1(C(C(C)N(C)C)=O)CCC(CNC(=O)C(C)CC(N)=O)C12CCC2 51759,c1(OC)ncccc1C(=O)NC(C)(C)CN(C(=O)Cn1ccc(C)n1)C 51760,c1(C(N2CC3(CC(CNC(CCSC)=O)OC3)C2)=O)cc2n(n1)CCCNC2=O 51761,c1(C(=O)NCCCNC(COC2(C)CCOCC2)=O)ccc2sc(O)nc2c1 51762,C(c1ccc(CN2CC3(CC3C(=O)NCC34CCN(CC3)C4)C2)cc1)=CC(=O)O 51763,Cc1cc(C(C)C(=O)N2CC(CNC(c3nc(C(C)(F)F)cs3)=O)C2)c(C)o1 51764,C1(NC(=O)Cc2ccc(Cl)cc2F)CN(C(=O)CC2CCOC2=O)CC1C1CC1 51765,c1(CC)nc(C)[nH]c1C(=O)NC(CNC(=O)C(C(C)C)SC)CC(C)C 51766,CC(C)(C(=O)NCC1CCCN(C(=O)CCOCC(F)(F)C(F)F)C1)C(F)(F)F 51767,C(N=c1ncc(CCOC)c[nH]1)C1CCC(C(C)OC)CC1 51768,N1(C(C(CC)CC)=O)CC2CCCC(N(C(=O)C(COC)N(C)C)C)C2C1 51769,c1(C(N(C2CCN(C(c3nnn(C)c3N)=O)C2)C)=O)coc2cc(F)cc(F)c12 51770,c1(OC)ncnc(OC)c1CN1CCCC1CC(=O)Nc1sccc1CO 51771,CN1CCN(C(=O)C(N2CCOC(c3ccc(F)cc3F)C2)=O)CC1C(C)(C)C 51772,CCCCCC(=O)NN(CCNC(=O)C(C(C)C)Oc1ccc(Cl)cc1)C(C)=O 51773,C1(C(N(C(C)C)C2CC2)=O)CCCN(C(C2C(c3cccc(Br)c3)C2(C)C)=O)C1 51774,CC(CC(=O)N1CC(C)C1C(=O)N=c1ccn(C(C)C)[nH]1)CC(C)(C)C 51775,C1(NC(c2c(C)nn[nH]2)=O)CCC2CC1CN2C(=O)CCCCCC#N 51776,c1(OC)cccc2c(CC(N3CC(NC(=O)Cc4cc[nH]n4)C(C)C3)=O)coc12 51777,C1(C(=O)NCc2ccc(C(N(CCC(N)=O)CC)=O)s2)CCCCCN1C 51778,C1(NC(c2c(C)ccs2)=O)CCCCN(C(c2cnc(C(C)(F)F)s2)=O)C1 51779,C1(NC(c2c(CCC)n[nH]c2)=O)CC2(CNC(=O)CC3CCOCC3)CC1CO2 51780,C(c1cn(C)nn1)=CC(N1C(CNC(c2c(C(C)C)scn2)=O)C=CC1)=O 51781,c1(CN(C)C(=O)NC2CCC3CCCC23)cccc(Br)c1F 51782,C(=O)(C1=CCC(F)(F)CC1)N1CC(C2(NC(c3cc(C)no3)=O)CC2)C1 51783,C#CCCC(=O)NCCn1ccc(C(=O)NCC2(SC)CC2)c1 51784,C1(CCNC(C=CCOCCOC)=O)CC(NC(=O)COCCCC)C1(C)C 51785,c1(NC(C2C(C=C)OCC2)=O)c(OC)cccc1C.c12nc(cn1C)NC2=O 51786,c1(CCN2CCCC(C(C)OC)C2)c(O)nc(=O)n(CCl)c1N.C(=O)(C(C)C(C)=O)OC 51787,C(=O)(CS(=O)c1ccc(Cl)cc1)NC1CC(N(C(=O)C(C)(F)F)C)C1 51788,C1(C(=O)NC2(C)CN(C(C3CCCN(C(N)=O)C3)=O)C2)CCS(=O)(=O)C1(C)C 51789,N1(C(C(=O)NCC=C)C(C)C)CCOC(C)(C(F)(F)F)C1 51790,C(C(F)(C(=O)NCCC1CCCCO1)C(C)C)NC(c1c(C)nsc1C)=O 51791,CCC(CCC(=O)NC1CC2(C1)CC2C(=O)N(C)CCOC)OC 51792,N1(C(C=Cc2n(C)cnc2)=O)CCC2CCC(C1)N2C(=O)CC1(C)CC1 51793,C12(NC(c3ncc(C(F)F)s3)=O)CCC(C1)N(C(c1ccncc1C(F)F)=O)C2 51794,C1(CNC(CC)=O)CCC2(CCN(C(c3ccccc3COC)=O)CC2)O1 51795,CON1CC(C(=O)NCC2(O)CCN(C(=O)Cc3ccn(C)n3)C2)CC1=O 51796,C12(CNC(CCc3onc(CSC)n3)=O)CCCN(C(=O)COC(C)C)C1C2 51797,c1(C)cnc(Cl)c(N)c1.c12ccc(cc1)OO2.C12CCCN1C(=O)N(CC)C2.OC 51798,C1(NC(C)=O)CN(C(=O)CCc2cc(Cl)cc(Cl)c2)CC12CC2 51799,c1(CN(CCC(C)(C)C)C(c2ccccc2)C)nn(C)cc1Cl 51800,c1(NC(C23C(CN(C(c4n[nH]c(CC)c4F)=O)C2)C3)=O)ncc(C)cc1Br 51801,CCCCCC(O)C(C)C(=O)N1CCCC(CCNC(c2ccoc2Cl)=O)C1 51802,c1(C(=O)NCCC23C(CN(C(C4C(C)C4)=O)C2)CC3)cc2c(Cl)c(Cl)ccc2[nH]1 51803,CCCC(CC)C(=O)NC(CC(=O)NCC1(C#N)CCCCC1)C(C)OC 51804,n1(CC(C)CO)nc(-c2ccccc2)nc1CC1CC1(C)C 51805,c1(CNCC(c2ccc(C3CC3)cc2)(C)C)cc(F)cc(O)c1F 51806,Cc1cnn(CCC(=O)NCC(O)CNC(c2csc(Cl)c2)=O)c1 51807,C12(C(=O)NC(C)C(C)NC(c3cncn3C)=O)CC(CCO1)C2 51808,C1(CNC(C(c2cncnc2)C)=O)COC(C)(C)CN1C(c1ccoc1C)=O 51809,c1(N2C(C)CC(NC(=O)CCCc3ccccc3Cl)C2)cc(C(N)=O)nc(Cl)n1 51810,C12(SCC(N3CC(C)C(C)(CN=c4ccnc[nH]4)C3)=O)CC3CC(CC(C3)C1)C2 51811,c1(C(N2CCC(N(C(=O)CCC(F)F)CCC)C2)=O)ccc2c(c1)CCOC2 51812,c1(CC(N2CC3CC(NC(C4(COC5CC5)CC4)=O)C2C3)=O)c(Cl)cccc1Cl 51813,Cc1cc(CNC(=O)CC(C)NC(c2ccccn2)=O)cc(C#N)c1 51814,c1(CN(C(=O)C(C)OC2COC2)CCNC(CC=CC)=O)ccccc1 51815,N1(C(C2(C)CSC2)=O)CCC2(CC1)CC2C(=O)NCCCCc1cnc[nH]1 51816,C=C=CC(C)C(=O)N1CCOCC1C(=O)NCC(C)C(F)F 51817,c1(C(CN(c2nc(C3CC3)ns2)C)O)cccc([N+](=O)[O-])c1 51818,CC(CCCNC(=O)CCc1cnoc1)NC(=O)CSc1nncs1 51819,C1(NC(C2C(CC)C2)=O)CC2CC(NC(c3cc(Cn4cccn4)on3)=O)CC12 51820,c1(CCC(=O)NC23CC2CN(C(c2ccoc2Cl)=O)C3)nnc(O)nc1O 51821,Cc1ccc(O)cc1C(N1CCC(NC(=O)C=C2CCN(C)C2)C(F)C1)=O 51822,C#CC1(C(=O)NCC2CC(n3cccn3)C2)CCN(C(=O)C(CSC)OC)C1 51823,c1(C(N2CCN(C(c3c(CC)scn3)=O)C3C2C3)=O)cc2cccn2c(O)n1 51824,N1(C(C2N(C(CCCCC)=O)CSC2)=O)CCC2(CSC2)C1 51825,c1(C(C)NC(=O)NC(CC2CC(F)(F)C2)CO)nc2c(o1)CCSC2 51826,c1(OCC)c(C)[nH]c2ccc(OCC3CC3)cc12.C12C(C1C1CNC1)C(=O)N2 51827,CCC(CC(=O)NCC1CC1C(=O)NCC1CC2(CCC2O)C1)CC(C)C 51828,N1(C(C2(C(N(C)C)=O)CC2)=O)CC(NC(c2ccn(C(F)(F)F)n2)=O)CC(F)C1 51829,Cc1cnccc1-c1cn(CCCN(C(=O)CC2CC3CCC2O3)C2CC2)nn1 51830,C#Cc1cccc(OCC(=O)NC2CCOCC2NC(=O)CC(=O)N(C)C)c1 51831,c1(C(N2CC(CN(C)C(C3CCCS3)=O)C2)=O)csc2nccn12 51832,C(C1=CCN(C(c2cc(CCCO)on2)=O)CC1)NC(=O)C(F)=CC1CC1 51833,C1(c2nnnn2C)(NCC(c2ccc(OC)cc2)(C)OC)CCC(C)(C)C1 51834,C1(NC(c2cc(C)nc(C)c2)=O)CN(C(=O)CC2CCCN(C)C2)CC(C)(C)C1 51835,C(C(C)(C(=O)N1CC2C(C)C2C1)NC(c1cccc(CC#N)c1)=O)SC 51836,c1(C(=O)NCCCCCO)nc2ccc(Br)cn2c1F 51837,C(CC(C)C)(C(=O)NCC1CCCN(C(=O)Cc2cocn2)CC1)OC 51838,C1(CC)CN(C(C2(C)C=CCC2)=O)CCN1C(=O)COc1cc(C)on1 51839,C12(C(N(C3CCCCC3)C(CC)C)=O)CC(CN(C(c3cnccc3C)=O)C1)C2 51840,N1(C(C2C(CNC(C3CC4(CCC4)C3)=O)CCO2)=O)CCC(=C(F)F)CC1 51841,C=CCCC(C(=O)Nc1cn(C)nc1OCC)NC(=O)Cc1ccccc1F 51842,Nc1cc(C(N2CC3CC2C3NC(=O)CC(O)C2CCCC2)=O)c(Cl)c(F)c1F 51843,Cc1ncnc(N2CCC(CNC(=O)COC(F)(F)F)C2)c1Br 51844,c1(C(=O)NC(CC)(C)CNC(=O)COCP(C)(C)=O)ccc(Br)cc1 51845,N(C(=NCC(C)C)N1CCC(CC(C)C)C1)CC(c1ccc(F)cc1)OC 51846,c1(C(N(C)CC2N(C(C(C)NC(C)=O)=O)CCC2)=O)c(C)nc2cccnn12 51847,c1(OC)cncc(C(=O)NC2CN(C(=O)C(CO)N(C)C)CC2CC(C)(C)C)n1 51848,C(=O)(CC(C)CNC(C1CCOC1C1CC1)=O)NCC(CSC)OC 51849,N1(CC(N2CC(c3n(C)cnc3)C(NC(=O)CNC=O)C2)=O)CCC(=O)NC1=O 51850,N1(C(c2nc(Cl)sc2Cl)=O)CCN(C(C2CC3COCC3C2)=O)C2COCC12 51851,C(C(C(C)C(C)C)NC(=O)Cn1ccc(C)cc1=O)NC(C)=O 51852,C1(CC(=O)N(C2CCN(C(c3cnc4n3CCS4)=O)C2)C)CN2CCC1CC2 51853,n1(CC(=O)NCCN(CCC)C(C2CCC(=O)C2)=O)c(C)c(C)sc1=O 51854,C1(CNC(CNC(=O)OC)=O)CCCN(C(C2CCC(C)(C)C2)=O)C1 51855,C12(CNC(c3cc(C)sn3)=O)CC3CC(CC(C3)C1NC(C1CNC(=O)C1)=O)C2 51856,CC(CN=c1[nH]nco1)(C1CC1)NC(c1cc(S(N)(=O)=O)co1)=O 51857,CCC(CC)C(=O)NCc1nnn(C)c1C(N1CCCCC1C1CC1)=O 51858,C1(C(=O)NC(C2N(C(CCC(=O)NC)=O)CCCC2)C)C2(CCC2)C12CCC2 51859,C(=O)(C(C)N(CC(C)NC(=O)C(C)C1CC1)C)N(C1CC1)CC 51860,n1(CC)nc(C)cc1C(=O)NC(C)C(C)(C)NC(C1CNC(=O)C1)=O 51861,C1(CC(Cc2ccc(C)cc2)C)CCN(c2ncccn2)CC1C 51862,N(C1CCCn2ncnc21)C(C(C)(N(C(COC)=O)C)C1CC1)=O 51863,c1(C(=O)NCC(CNC(C(C)OCC)=O)OC)cc(Cl)c(Br)cc1C 51864,C(=O)(CC1=CCOCC1)NCC(CC)NC(C1CC(C)(C)OC1(C)C)=O 51865,N1(C(C(CC(C)=O)(C)C)=O)CCC2(CCCN2C(=O)CC2CCCC2C)C1 51866,N1(C(C=CC(=O)OCC)=O)CCCC2CCN(C(c3n[nH]c(C4CC4)n3)=O)CC12 51867,N1(C(=O)CCSc2ccccc2)CC2CC(C1)N(C(=O)C=C(Cl)Cl)C2 51868,C(C(C)(C)CC(=O)NC1CCOCC1NC(=O)CSCC(F)(F)F)OC 51869,C(C(C(=O)Nc1cnn(CCF)c1)C(C)(C)C)NC(c1c(C)n[nH]c1C)=O 51870,c1(N(C)C)ncc(Br)c(C(=O)NCC(C(C)C)NC(=O)CC2CC23CC3)n1 51871,N1(C(CC(N2CCCCC2=O)C)=O)CC2CN(C(C3C(C)(C)C3(C)C)=O)CC2C1 51872,c1(C(N2C(C(=O)NCC(CCC)C)CCCC2)=O)cc(C)cc(F)c1 51873,Cc1nc(CC(=O)NC2C=CCN(C(c3cc(C4CCOC4)[nH]n3)=O)C2)[nH]c1C 51874,CC1(C)CCC(C(=O)NC2COCC2CO)(NC(=O)CNc2cccnc2)C1 51875,N1(C(C(C)(C)N2CCOCC2)=O)CC2CC2(CNC(=O)C=CC(=O)NC2CC2)C1 51876,C1(C(=O)NCCN(CCC)C(c2ncsc2NC)=O)CCC(C2CC2)C1 51877,C1(C(=O)NCCC2CN(C(C3(C(C)(C)C)CCCC3)=O)C2)COC2CCCCC12 51878,N1(C(c2c(C(=O)OCC)cccc2)=O)CC2CC1CN2C(=O)Cn1nnc(C)n1 51879,c1(C(=O)NC(C)CNC(=O)CN2CCSCC2)ccc(SCc2cnc[nH]2)cc1 51880,N1(C(c2ccn(C(F)F)n2)C(=O)NC)CCCC(O)(C(C)C)C1 51881,c1(OC)c(C)ccc(C(=O)NC2COCCC2NC(=O)CCc2cnoc2)c1F 51882,CC1CCCc2ncc(C(=O)NC3CC34CCN(C(=O)Cc3cnoc3)CC4)n21 51883,C1(CC)(NC(C2CCCN(CC(C)C)C2)=O)CCCN(C(=O)Cn2cnnn2)C1 51884,C12(CNC(C3(C#C)CCC3)=O)CCC(CC1)N(C(c1ccoc1)=O)C2 51885,c1(CN(C(C2CC23CCOC3)C(=O)NC2COC2)CC)ccc(OC)cc1Br 51886,C1(C(N(CCN(C(c2cnn(CCF)c2)=O)CC)CC)=O)CC(NC)CCO1 51887,S(=O)(=O)(c1ccc2c3c(cccc13)CC2)NCC(c1cccc(Cl)c1)C 51888,c1(C(=O)NCC(CCOC)NC(c2cc(C)ns2)=O)nccc2cc[nH]c12 51889,C1(CNC(c2cccnc2)=O)CN(C(=O)CCc2ccccc2O)CC1(F)F 51890,c1(CCCNC(N2CCCC2c2ncno2)=O)cccc(Br)c1 51891,N1(C(CC2(COC)CCCC2)=O)CC2CCN(C(=O)Cc3csc(C)n3)CC12 51892,Cc1ccc(C(N2CCC(CN(C)C(C3COCCO3)=O)C2)=O)cc1CO 51893,N1(C(CCCCCCC)=O)CCN(C(C2CCc3cncn3C2)=O)CC2(CC2)C1 51894,CCC(CCC(=O)OC)N=C(NCCCCC(C)(F)F)NCC(C)(C)C 51895,C1(NC(c2ncn(CC)c2)=O)CCC(N(C(=O)COc2cn[nH]c2)C)CC1 51896,C1(C(=O)NCCN(C(=O)C(F)C2CCOC2)CCOC)CCC=CCCC1 51897,Cc1cccc(C(=O)NC(CNC(=O)CN2CCOCC2=O)C(C)C)c1F 51898,c1(NC(CC2OCCN(C(C3C(C(=O)OCC)CC3)=O)C2)=O)ccc(C)nc1C 51899,c1(-c2ccc(C)c(O)c2)cc(C(=O)N=c2[nH]c(Cl)ncc2C)c2[nH]ccc2c1 51900,Cc1csc(C(N2CCCCC2C(C)(C)CNC(c2ccnnc2C)=O)=O)c1C 51901,CC(N=c1nn[nH]n1C)C1CCCCN1C(c1c(Cl)cnn1C)=O 51902,N1(C(CCCC=C)=O)CC2CC(C1)C(CO)C2NC(=O)CSC1CCS(=O)(=O)C1 51903,N1(C(C(C=C=C)C)=O)CCC(CC(=O)NCC(C2CCCC2)C)C1(C)C 51904,CCC(CC(=O)N(CCCN(C)C(C1CCC(C(=O)OCC)CC1)=O)C)OC 51905,CN1CCC(NC(N2CCOC(CO)C2)=O)C(c2ccccc2)C1 51906,N1(CC(c2nccs2)=O)CC(n2cc(C(c3ccccc3)O)nn2)C(O)C1 51907,C1(C(=O)NC2CC(CCNC(c3ncncc3Cl)=O)C2)CC2(CCCCC2)CO1 51908,c1(OC)ccsc1C(=O)NCC1CCCC1C(=O)NOCc1nc[nH]n1 51909,c1(C(N2CCC(CNC(C3CCC34CCC4)=O)C2)=O)cccc(C#CCO)c1 51910,c1(C(=O)NCC2C(C)CCN(C(=O)CSC(C)(C)C)C2)cc2ccccn2n1 51911,C1(NC(c2cc(CCC)[nH]n2)=O)CCN(C(C2OC3CCC2CC3)=O)CC(O)C1 51912,C1(CNC(C=CSC)=O)CCN(C(=O)CCc2ccccn2)CC1(F)F 51913,c1(C(=O)NC(c2ccccc2F)CNC(C=CCOC)=O)nccnc1O 51914,CC1CC(C(N2CCN(C(=O)CCNc3ncccn3)CC2)=O)CC(=O)N1 51915,N1(C(CC(C)(C)OC)=O)CCC2CCCC12C(N1CC2C=CC1CC2)=O 51916,C1(NC(C2(C)CCOCC2)=O)CCC2(CC1)CCN(C(=O)C(F)F)CC2 51917,c1(C(N2CCOCC(CNC(COCC=C)=O)C2)=O)ncc2ccccn12 51918,CC1(COC(c2ccn(C3CCCCC3)n2)=O)CCC(F)(F)CC1 51919,CC(C)C(N=[N+]=[N-])C(=O)N1CCC(C)(C)C1C(=O)NC1CC2CC1CC2(C)O 51920,C1(CNC(Cc2c(C)nc(C)s2)=O)CC2(CO1)CN(C(=O)C(C)CS(C)(=O)=O)C2 51921,N1(C(C=Cc2ccc(C)s2)=O)CCCCCC1CNC(=O)CC1CC=CCN1C 51922,CCCC(O)CC(=O)N(CCNC(=O)C(F)C(C)(C)O)CCOC 51923,C=CCN=c1ccc(S(=O)(=O)N2CCCCC2c2ncc(Br)cn2)c[nH]1 51924,N1(C(c2cc(OC)ncn2)=O)CC(NC(=O)COC(F)(F)F)CC1(C)C 51925,C1(CC(=O)OCC2(C)CCCC2O)(NC(=O)OC(C)(C)C)CCCCC1 51926,CCC(CNC(c1cc(C#N)oc1C)=O)(CC)C(=O)NC12CCCCC1C2 51927,CCCCS(=O)(=O)CC(=O)NCC(CO)NC(c1csc(C)n1)=O 51928,Cc1ccc(C)c(C(=O)NC2CCCC2(C)NC(=O)CC2CCCO2)n1 51929,C(=O)(C1=CS(=O)(=O)CCC1)N1CCN(C2CCN(C(C(C=C)CC)=O)C2)CC1 51930,N1(C(CSc2ccc(C)cc2C)=O)CC(CNC(=O)CC#N)C2(CCC2)C1 51931,Cc1noc(C(C)C)c1C(=O)NCCC1CCN(C(=O)CC2CC2C)CC1 51932,C(C(=O)NC(C(=O)N(C)CC1CCOC1C)C1CCOC1)(C(C)(C)C)OC 51933,N1(C(C(C)=CC=C)=O)CCC(C(=O)NCc2ncsn2)=C(F)C1 51934,c1(C(N(C(C)C(=O)N(CCC(=O)NC2CC2)C)CCC)=O)cnc(C)o1 51935,C(C(C)(C1CC1)NC(=O)CNS(C)(=O)=O)NC(COC(CC)C)=O 51936,c1(COC)csc(C(C(=O)NCC(F)F)N(C)Cc2ccsc2)c1 51937,Cc1cc(C)n(CCC(N2CC3CC2C3NC(c2ccc(C(F)F)cn2)=O)=O)n1 51938,c1(NC(=O)CC2CCCC2C(N2CCCC2C2CCCOC2)=O)ncccc1O 51939,C1(NC(=O)COc2ccsn2)CC(F)(F)CC1NC(c1ccc[nH]1)=O 51940,Cc1cc(NC(=O)N(CC(C)C)Cc2ccccc2Cl)ccc1-c1ccncc1 51941,C#CC1CC2CCC1N(C(=O)C=CCN(C)CCOCCSC)C2 51942,Cc1nsc(CNC(c2nnnn2CCN2CCOCC2)(C2CC=CC2)C)n1 51943,C1(NC(=O)C=CCOc2ccccc2)(CO)CCCN(C(=O)C(C)OC2CC2)C1 51944,C1(C(=O)NC2(CC#C)CC2)C=CCN1C(C1CC(n2cccn2)C1)=O 51945,c1(CC)nc(C)c(C(=O)NC(C)CCN(C(=O)COCC2CCCO2)C)s1 51946,C(C1COc2ccccc21)NC(NC(c1cccs1)C)=NCCF 51947,C(=O)(CC(=O)N=c1ccn(C2COC2)[nH]1)NCCN1CCN(C)CC1 51948,c1(OC)ccc2c(c1)CC(C(=O)NC1CCCC1NC(C1(CCO)CC1)=O)CO2 51949,CCCC(C)(O)C(=O)N1CC(NC(c2ccc(CC)c(F)c2)=O)C1 51950,C1(C(=O)NC2CC(CCNC(c3cc(C4CCC4)no3)=O)C2)CC2(C1)OCCO2 51951,C12(C(N(CCNC(c3nn(CC)nc3C)=O)C)=O)CCC(C(F)F)(CC1)C2 51952,c1(C(=O)NCC=CCNC(c2occ(C)c2C)=O)c(O)cc(=O)n2c1CCCC2 51953,N1(C(C(C)NC(CN(C(C)C)C)=O)=O)CCC(N(C)C)C(C)C1 51954,c1(C(c2cc[n+]([O-])cc2)=O)cnc(Cl)[nH]c1=NC1CC2CCC1N(C(C1CCC1)=O)C2 51955,c1(C(N2CC(C=C)(CC(=O)NC3(C)CCCC3O)C2)=O)nccc(C)c1F 51956,c1(C(=O)NC2CN(C(C3CC4(CC(OC)C4)C3)=O)C2)c(Br)ccc(F)c1C 51957,C1(CNC(c2cnc(CC(C)(C)C)s2)=O)CN(C(C2CSCCS2)=O)CC1O 51958,c1(C(=O)NCCCNC(=O)C(Cl)=CCl)cccc(-c2cccs2)n1 51959,C(=O)(CCCCCC(C)C)NCC1N(C(c2c(C)ccc(Cl)c2)=O)CC(F)C1 51960,c1(CCNC(=O)NC2(C(F)F)CCC2)ccc2c(c1)OCCO2 51961,C1(CC(=O)N(C(C)C(=O)NCCn2cnnc2C)CC)CCC(C)CO1 51962,CCC(C)C(O)C(=O)N1CCN(C(=O)C(C)(C)c2ccno2)CC1Cc1cn[nH]c1 51963,N1(C(C=NOC)=O)CCC(CNC(C2CCOC2C(C)C)=O)CC1 51964,CCC(C(=O)N1CCN(C(c2ccnnc2O)=O)C(CO)C1)C(C)(C)CC 51965,CC1(C=CC(=O)N(C2CCCN(C(=O)CC3CC34CC4)C2)CCO)CCOCC1 51966,S(=O)(=O)(CCCCS(N)(=O)=O)N1CCCC(C(C)(O)CN)C1 51967,C(=O)(C(C)Cc1ccnn1C)N(C1CN(C(C2(SC)CC2)=O)C1)C 51968,C(=O)(C(F)(CNC(c1ccccc1C1CC1)=O)C(C)C)N(CC=C)CC 51969,C1(C(=O)NC(CC)CC(F)(F)F)CCC2(CN(C(c3ccccc3)=O)C2)O1 51970,c1(-n2c(COCC(C)C)nc(-c3cncc(F)c3)n2)ccc(Cl)c(Cl)c1 51971,CCC(CC)C(C(=O)NC1(C(=O)NCC(C)CC2CC2)CSC1)OC 51972,C(N=c1[nH]cnc(NCc2ccc(Cl)c(F)c2F)c1C)c1cc(CC)no1 51973,c1(CC)nc2c(C(=O)NCC(C)(CO)NC(=O)C(C)C3CC3)ccnc2[nH]1 51974,CC1(C)CC(NC(c2cc(O)cc(Br)c2)=O)CN1C(c1ccnnc1O)=O 51975,CCC(CN=c1[nH]c(=NCCC=CBr)[nH]c2c(F)cccc12)n1cccn1 51976,Cc1nnc2c(C(N3CCCOC(CNC(=O)C(C)(C)C)C3)=O)cccn12 51977,C1(C(C(=O)NC(c2cccnc2)C(=O)N(C2(CC)CC2)C)C)CCOCC1 51978,c1(OC(C)C)cncc(C(=O)NCCCC(C)(C)NC(c2ccco2)=O)c1 51979,c1(N)cc(Cl)c(Br)c(Cl)c1.CC1C(C(=O)NOCC(O)CO)C1C 51980,c1(C(=O)NC(C2N(C(C3C(CC)C3)=O)CCC2)C)cc2c(nc1O)CCOC2 51981,N1(C(C=CC=CC)=O)CCC2(C(=O)NCc3cnccc3C)CCCC12 51982,C(c1ccnn1C)=CC(=O)NC(C(=O)NC(c1n(CC)ncc1)C)c1ccco1 51983,c1(C(C)=O)ccc(C(=O)NCC2(O)CC(C(=O)NC(c3ccoc3)C)C2)o1 51984,CCCC(C(=O)NCC(CNC(=O)Cn1cnccc1=O)OC)c1ccccc1 51985,C1(C(=O)NCC(CSC)OC)CCC(O)CN1C(=O)Cc1nocc1C 51986,N1(C(C2N(CC)CCC2)=O)CC2CC(C(=O)NCc3cc(C)sc3C)(C2)C1 51987,C1(NC(c2cc(OC)n(C)n2)=O)CN(C(=O)CC2CCCS2(=O)=O)CCC1CO 51988,CC1CCN(C(=O)Cc2ccc(Br)o2)CC1NC(=O)Cc1ccccc1CO 51989,c1(CN(C)C(=O)NCc2cncc(Cl)c2)nc2c(s1)CCCC2 51990,c1(COC)ccc(C(N2CC(NC(=O)CC3COC(=O)C3)CC2C)=O)cc1 51991,c1(C(C)C)cccnc1CN1CC(F)(c2ccccc2)C1 51992,CC(CC(F)F)C(=O)N(CCCCCCNC(C1(F)CCC1)=O)C 51993,C12(C(N3CCCC(CCC(=O)N(C)CCC4CCCC4)C3)=O)CCCC1C2(F)F 51994,n1(CC(=O)NC(c2ccccn2)(C)C)cc(C#N)c(O)nc1=O 51995,C(=O)(C(C)(C)C(C1CC1)NC(C1CC(=O)NO1)=O)OC 51996,Cc1c(C(=O)NCC2CC(CNC(=O)CSC(F)F)CO2)sc2ccc(F)cc12 51997,C(=O)(C(C)(C)C(=O)NCC(O)CN(C(=O)CCn1cc[nH]c(=O)c1=O)C)OC 51998,C1(CC=C)(NC(C2CC2(C)C)=O)CCN(C(=O)Cc2c[nH]ccc2=O)C1 51999,C1(F)(C(=O)NCCC2(O)CCN(C(C(C)SC)=O)C2)CC2(CCC2)C1 52000,c1(CC(=O)NCC2CC(NC(CCP(C)(C)=O)=O)C2)ccc2nsnc2c1 52001,c1(C(N2CCC(C)(CNC(C(C)P(C)(C)=O)=O)C2)=O)cccc2cc(O)ccc12 52002,N1(C(CCCCC)=O)CCN(C(=O)C(C)OC2CCCCC2)CC1CC(F)F 52003,CC1(C)CCC=C1C(=O)NCn1ccc(=O)n(Cc2ccccc2)c1=O.C1CN1 52004,C(=O)(CCCCCCCCCO)NCC1C(C)(C)CN(C(C2C=CCCC2)=O)C1 52005,Cc1nc(N2CCC(NC(=O)C(C3CCCO3)C3CC3)CC2C)cc(C#N)n1 52006,c1(COCC(=O)N(C)CC2C3CN(C(=O)C=CCF)CC23)ccc2c(c1)OCO2 52007,C1(O)(CNC(C(CCOC)OC)=O)CCCN(C(=O)Cc2cnc(C)s2)CC1 52008,c1(CC(=O)NCC=CCNC(=O)CCCCC2CC2)c[nH]c2ncccc12 52009,c1(C(=O)NCC2C(NC(COCC)=O)C2)cc(OC)c(OC)cc1N 52010,N1(C(c2cc(C)cc(OC)c2N)=O)CC2CC(C1)CN(C(C1CC1OC)=O)C2 52011,CCCCCC(O)C(=O)N1CCCC1Cn1cc(CNC(C2(F)CC2)=O)nn1 52012,N1(C(CC=CCC)=O)CCOC2(CCN(Cc3ccc(F)c(O)c3F)CC2)C1 52013,c1(CN2CCC3(C(NC(Cc4cn(CC)nc4)=O)C3)C2)cn2ccccc2n1 52014,N1(C(=O)CC(F)F)CCN(C2CCC(NC(=O)C(F)C3CC3)CC2)CC1 52015,CCC(O)CC(=O)NCC1CCC(NC(=O)CC2CSC2)CC1 52016,CCCC(CCCNC(c1ccc(=O)n(C)c1)=O)NC(c1sc(C)cc1C)=O 52017,c1(C(N(CC(C)NC(c2cc(CC)[nH]n2)=O)C)=O)ccc2cnsc2c1 52018,N1(CCN(C(=O)CCc2ccc(CO)cc2)C)CCN(C(=O)CC2(C)CC2)CC1 52019,C(=O)(C1=NN(C)C(=O)CC1)NCC(CC(=O)NC1CC(OC(C)C)C1)C1CCC1 52020,CC(C)(CO)C(=O)NC1(C)CCN(C(=O)COc2cccc(Br)c2)C1 52021,N1(C(C(c2ccc(Cl)cc2)C)=O)CC(NC(=O)C=CC(N)=O)Cc2ccccc21 52022,C1(C(=O)NC23CN(C(C(n4c(C)cc(C)n4)C)=O)C(C2)C3)CCn2ncnc2C1 52023,C1(CNC(Cn2c(C(C)C)ncc2)=O)CC2CCC1N(C(=O)Cc1cnns1)C2 52024,N1(C(Cc2c(Br)cn(CC)n2)=O)CC(C2(NC(=O)C3=CCCS3)CC2)C1 52025,CC1CCOCC1C(=O)NCC1(NC(c2cccc(N(C)C)n2)=O)CCC1C 52026,C=CC1(CNC(C2(C)CC(O)CN2C(=O)C(C)c2cccs2)=O)CCOCC1 52027,C1(C(N2CCC(NC(=O)CCCCCF)C2)=O)(COC)CCCNS1(=O)=O 52028,C1(C2(O)CCC2)(C(=O)NCCCCNC(c2cnc(CCCC)s2)=O)CC1 52029,n1(CC(=O)NCCc2ncc(C(=O)O)s2)cc(C(O)C2CC2)nn1 52030,C1(COC)CC(O)CN1C(C1COCCC1NC(c1cc(Cl)n[nH]1)=O)=O 52031,C1(C(N2CC(NC(C=C(C)C(F)F)=O)C3(C2)CC3)=O)CCOCC12CCCCC2 52032,N1(C(c2c(C)nc(C3CC3)s2)=O)CCC(CNC(c2ccc(Cl)nn2)=O)C(C)C1 52033,C(=O)(C1CCCc2ncnn21)N1CCN(C(c2[nH]nnc2C2CC2)=O)CC(C)C1 52034,N1(C(c2c(C)c[nH]n2)=O)CCC(O)C(C(=O)NCc2ccccn2)C1 52035,c1(OC)ncc(CNC(=O)C(C2CCC(=O)N2)C)s1 52036,Cc1cc(C(=O)NC23CCCN(C(c4ccsn4)=O)C2C3)ccc1Br 52037,c1(C2C(C(=O)NC(CNC(c3c(C)nc(CC)s3)=O)C)C2)ccc2c(c1)OCO2 52038,N1(C(CCC(=O)NCCC)=O)CCN(C)C(C(=O)Nc2ncc(C(=O)OC)s2)C1 52039,c1(C(=O)NC2CCCC(N(C(=O)Cc3ccoc3)C)C2)ccc2ccn(C)c2c1 52040,N1(C(CC)CSC)CCc2c[nH]c(=N)nc2C1 52041,c1(C(=O)NC2CCC(NC(=O)C(F)=CC3CC3)CC2)cc2c(cn1)OCCC2 52042,N1(C(c2cnc(N)c([N+](=O)[O-])c2)=O)CCCC2(CCCCC2NC(=O)CCF)C1 52043,C1(CNC(c2n(C=C)ncc2)=O)CC2CCC1N2C(C1SCCCS1)=O 52044,C1(NC(=O)CCc2cncnc2)CC2CC(C1)N(C(=O)CN1C(=O)CNC1=O)C2 52045,C(C(O)CCNC(C1(n2nccn2)CC1)=O)NC(COCCSC)=O 52046,c1(C(=O)NC(CNC(C(c2ccc(CC)cc2)C)=O)C2CC2)cc(C)cc(N)c1 52047,N1(C(C(C(CC)CC)C)=O)CCC(NC(=O)C(C)C(=O)OC)C2(CCC2)C1 52048,CC1CN(C(C2(C)CCCOC2)=O)CCC1CNC(c1ccc(F)cc1F)=O 52049,C1(CNC(C(C)NC(N)=O)=O)CN(C(=O)CC2CC(F)(F)C2)CCC1(C)C 52050,N1(C(C2CC(C#N)(OC)C2)=O)CC(NC(c2cnc(N(C)C)s2)=O)C2(CCC2)C1 52051,C=C(C)C(O)CC(=O)NC1CN(C(c2cc(OC)ccc2F)=O)CC1C 52052,CN1CC(C(N2CCCC(C(=O)Nc3nccc(CO)n3)C2)=O)CC1=O 52053,Cc1ncc(C(=O)NC2CC(CNC(c3ccc(F)cc3)=O)CC2O)n1C 52054,Cc1cc(Cl)ncc1CC(=O)NC1CCC(CNC(=O)CC2CCC3CC23)CC1 52055,CC1(C(=O)NCCC2CC(NC(=O)CC3CCSCC3)C2)CCCC1 52056,c1(-n2c(C(CC=C)CC)nc(-c3occc3C)n2)ccc(C)c(F)c1 52057,C=C=CCCC(=O)N1CC(CNC(C2CN(C)C(=O)N2)=O)C1 52058,c1(C(=O)NCC(C)CNC(c2nnn3c2CCC3)=O)nccc2ccncc12 52059,c1(C(N2C(CCNC(C(CC#C)O)=O)CSCC2)=O)cccc(F)c1C 52060,Cc1nc(CCC(=O)NC2CCCC2NC(c2cc(F)n(C)n2)=O)[nH]c1C 52061,CCC(F)(F)C(=O)NCC1CC(NC(c2cnc(C)nc2)=O)C1 52062,c1(NC(=O)C2=CCN(C(=O)OC(C)(C)C)C2)cc(Cl)cc([N+](=O)[O-])c1 52063,CC(C)(C)C(C#N)C(=O)N1CC=CC(C(=O)Nc2cccc(F)c2)C1 52064,C1(NC(C2(CCNC(c3c(C(C)C)onc3)=O)CCC2)=O)CCn2nccc2C1 52065,C(=O)(C1=NOC2COCC12)NC(C(C)C)CCN(C(=O)CCC1CC(F)(F)C1)C 52066,C1(C(=O)NCC(C=C)(F)F)CC2(CCO2)C1 52067,N1(C(CC(C)O)=O)CCCCC(N(C)C(c2cc(C(F)(F)F)ccn2)=O)C1 52068,C1(CC(=O)NC(c2c(C)nns2)C)CC2(CC2)CN1C(c1nnn(C)c1N)=O 52069,C(=O)(C(C)(O)C(C)(C)C)NCC1CC2(CC(NC(C(CC)CCOC)=O)C2)C1 52070,c1(N2CCC(CCNC(C(C)c3ccsc3)=O)C2)cc(=O)n(C)cn1 52071,C1(C(=O)OCC)CCN(C(=O)CN(C)CCOC(C)=O)CC1(C)C 52072,C1(C(=O)NCC2OCCN(C(C(C=C)O)=O)C2)CC2CCC1CC2 52073,Cc1nc(NCCN2CC3CCC3(CO)C2)cc(N2CCC(CCO)C2)n1 52074,CC(C)(CNC(=O)NCC1CCC12CCCO2)CS(C)(=O)=O 52075,c1(CC(=O)NC(C)C(C)(C)NC(=O)CCCc2nccs2)ccc2c[nH]nc2c1 52076,c1(C(=O)NC(C(N2CCCC(C=C)C2)=O)C2CCOC2)coc2ccccc12 52077,C1(C(=O)NC2CC(O)(Cc3cn(CCOCC)nn3)C2)CCOC(C)(C(=O)O)C1 52078,N1(C(=O)N(C(C)C)Cc2cccnc2)CCC(C)(Nc2cncc(C)c2)CC1 52079,CC1CN(C(=O)CC2CC2CNC(=O)C=Cc2cccnc2)CCS1=O 52080,c1(OC)ccc(NC2(c3nnnn3CC)CCOCC2C)cc1OC(C)C 52081,c1(C(N2CCCC(O)(CNC(C(=O)NCC)=O)C2)=O)cnc2cc(OC)ccn12 52082,C1(C(=O)NCC(CCOC)NC(=O)Cc2ccc(N)cn2)CCc2nn[nH]c2C1 52083,c1(C(=O)NC2C(C)(CNC(COCCC)=O)CCC2)sc2nccnc2c1NC 52084,C(=O)(C1=CCCOCC1)N1C(C)CC(C(=O)NCCCCCCF)CC1 52085,C1(NC(C2CN(CC)C(=O)N2)=O)CN(C(c2cocn2)=O)CCC1F 52086,C(=O)(C1CCc2ccccc21)N1CCC(N=[N+]=[N-])(C(=O)NCC(C#C)C(C)C)C1 52087,N1(CC)CCOCC1C(=O)NCCCCC(=O)NCCC1CCCN(C)C1 52088,C1(C(=O)NC(C)(CO)C2CCC2)CCN(C(=O)C(CO)NC(N)=O)C(C)(C)C1 52089,CC1OCCCC1C(=O)NC1CCC(C(=O)NCC(O)CN(C)C)CC1 52090,C(c1ccccc1)=CC(N1CC(CCCCNC(CC2C(CC)C2(C)C)=O)C1)=O 52091,C(=O)(C(O)C(C)(C)C)N1CCC(O)(CN(C(CCOCCC)=O)C)C1 52092,Cn1cc2c(n1)CCCC2C(=O)NC1CC(F)CN(C(=O)CC(C2CC2)C2CC2)C1 52093,C(=O)(C1=CCCOCC1)N1CC(CCOC)N(C(c2nc(C)ccc2F)=O)CC1 52094,CC1(C)CCC=C1C(=O)NC1CCN(C(=O)Cc2ccccc2Br)C1 52095,C(CC(F)(F)F)N(C)C(C1(CNC(=O)CC2CCOCC2)CC1)=O 52096,Cc1cccc(SN)c1.N1(C(COC)=O)CCC(c2cn(CCC3CC3)nn2)CC1 52097,c1(N2CC(C(C)NC(c3csnn3)=O)C2)c(F)cc([N+](=O)[O-])cc1F 52098,c1(C(=O)NCCCCNC(C(N)=O)=O)ncccc1Br 52099,c1(C2(CNC(c3n(CCCC)nnn3)(C)CCOCC)CC2)cc(C)cc(F)c1 52100,C1(NC(=O)COC(F)(F)F)CN(C(c2cnn[nH]2)=O)C2CCCCC12 52101,c1(C(=O)NC2(CNC(C(CSC)C)=O)CCCCC2)[nH]cc2c1CCS2(=O)=O 52102,c1(CC(=O)NC2CN(C(C(C)=C3CCC3)=O)CC(C)C2)ccc(S(N)(=O)=O)cc1 52103,CC1CN(C(=O)CSc2nnnn2C2CC2)CC1NC(C1(C)CCC(=O)C1)=O 52104,C1(CNC(C2(CC(C)C)CC2)=O)CN(C(c2csnc2Cl)=O)CC1C 52105,CC(CCN(C)C)C(=O)NCC1C2CN(C(=O)C(C)(C)N(C)C)CC12 52106,c1(C(=O)NCC(C)N(C(=O)C(C2CCCCC2)F)C)cscc1C(N)=O 52107,c1(C(N(CCC)CCNC(C2(CC)CNC(=O)C2)=O)=O)cc2cscc2s1 52108,CC1CN(C(c2ncncc2Cl)=O)CC(C)N1C(=O)CCC1CCOCC1 52109,c1(C(=O)NCC2(C)CCC(NC(c3cccnc3Cl)=O)C2)cncc([N+](=O)[O-])c1 52110,C1(C(=O)NC2(CNC(C3(CN(C)C)CC3)=O)CCOCC2)Cc2nncn2C1 52111,C1(NC(c2cccc(-n3cccn3)c2)=O)CC(F)CN(C(c2n[nH]cc2Cl)=O)C1 52112,c1(C(N2CCC(CNC(C(C)Oc3ccc(C)cc3)=O)C2)=O)c(C)[nH]c(C)c1C 52113,CCC(C)(CNC(C1(NC(=O)CC2CCCCO2)CC1)=O)OC 52114,C=CCCC(CC(C)C)C(=O)NCCN(C(=O)CCC1(C)CC1)C(C)C 52115,c1(C(N2CCN(C(COCCC#C)=O)C(C(C)C)C2)=O)cc(Cl)cc2c1CCC2 52116,c1(C(N(CCCCCNC(C(CC=C)CC)=O)C)=O)ccc2c(c1)nc(C)n2C 52117,C(C1CN(C(=O)C(O)Cc2ccccc2)CC1C(=O)NCC(F)C1CCC1)=CC 52118,C1(c2cn(CCF)nn2)(C(=O)OC)CCN(C(c2ncc(Br)s2)=O)C1 52119,c1(C(=O)NCCOC2CCN(C(C3(CCCC)CCCC3)=O)C2)nccnc1C 52120,C1(CCNC(C2=CC(C)(C)C2)=O)CCN(C(C2CCCO2)=O)CCC1(F)F 52121,CCC(C(=O)OCC)C(=O)N(CCC(=O)NCc1nc(C(N)=O)co1)OC 52122,C(C1CCN(C(c2nccn2C)=O)CC1)=CC(=O)NCc1c(C)cnn1C 52123,c1(CN(C(CC)CC)Cc2nc(C)c(C)s2)nc(C)c(C)nc1C 52124,CN1CCN(C(C2CCSC2)=O)CC1CNC(C1CC(F)(CO)C1)=O 52125,C1(C(=O)NCC(C)(O)CNC(c2c[nH]nc2C2CCOCC2)=O)(OC)CCCC1 52126,c1(CCNC(=O)NCC2CCCCS2)ccc(Cl)cc1 52127,N1(C(c2nc(C(=O)NCc3ccc(Br)cc3)sc2)=O)CC2CCC1CO2 52128,c1(CNC(=O)CCOC2CC2)cnn2c1CN(C(=O)CC13CC(C1)C3)CC2 52129,C(=O)(C(C)(C)CS(C)(=O)=O)N1CC(NC(=O)C(C)(C)N2CCCCC2)CC(C)C1 52130,N1(CC=CC=C)CCCC(C(=O)NCCSc2noc(C)n2)CC1 52131,CN1CCN(C(=O)CCc2ncnn2C)C(C(=O)NCc2cc(C3CC3)no2)C1 52132,N1(C(c2cc(C)n(CCO)n2)=O)CC2(CC(NC(=O)CCCC(C)O)CO2)C1 52133,Cc1cc(C(=O)NCC(O)CN(C(=O)Cc2c(C)noc2C)C)sc1Br 52134,C(C)(C(C)C(=O)NCCSCC1CCC1)NC(C1(C(C)C)CCC1)=O 52135,C(CC(C(C)(C)C)NC(c1ncccc1Cl)=O)N(C)C(c1cc(F)ccc1F)=O 52136,C1(C(=O)N(C2CCCOC2)C)(NC(C=C(C)C2CC2)=O)CCCCC1 52137,C=CC1(C(N2CCCC(C)C2CO)=O)CCN(C(c2ccc(C)c(F)c2)=O)C1 52138,C1(CC=C)(NC(=O)CSCCCC)CCN(C(c2cc(Cl)c(Cl)[nH]2)=O)C1 52139,N1(C(c2cc(C#N)no2)=O)CCOC2CN(C(=O)COc3cccc(F)n3)CC12 52140,O(NC(=O)CN=c1nc(CC)cc(C)[nH]1)CCSC(F)F 52141,CC(C)(C)C(CO)C(=O)NC1(NCCNC(=O)CCCCCO)CCOCC1 52142,c1(C(=O)NCCC2CCN(C(C3CC3F)=O)C2)csc2cccc(F)c12 52143,C1(C(=O)NCC=CCNC(c2c(C)c[nH]n2)=O)CCc2nnc(O)n2C1 52144,CC(O)C(C(=O)NCC1(NC(c2csc(C3CC3)n2)=O)CCCCC1)N(C)C 52145,c1(C(N2CC3(CN(C(C)=O)C3)C2)=O)cc2cc[nH]c(=O)c2s1 52146,N1(C(C2ON=C(CC)C2)=O)CC(OC)C(OC)C1CNC(=O)COc1ccsc1 52147,c1(OC)c(Cl)cc(NCCOC(C2CCC23CC3)c2nnnn2C)cc1Cl 52148,CC1CN(C(=O)C=CC2COC(C)(C)O2)CCN1C(c1cncs1)=O 52149,C(=O)(CC(F)(F)C(F)F)N1CCN(CC(=O)N(C)CCN(C2CCSC2)C)CC1 52150,C12CC(C)N1C2=O.n1(C2(CNC(COCCC)=O)CC2)cccn1 52151,C1(C(=O)NCCCCN2CCCC2)CN(C(C2COCOC2)=O)CC12CCC2 52152,C(N=c1cc[nH]cc1S(=O)(=O)NCC1CCCN1S(C)(=O)=O)C1CCC(C)O1 52153,c1(C(N(CC(CC)NC(C2(COC)CC(=O)C2)=O)C)=O)nc(O)c(C)s1 52154,CCS(=O)(=O)CC(C)NC(c1cc(N(C)C)ccc1C)c1nnnn1CC(F)F 52155,C(=O)(C1CCc2cccnc21)N1CC(CNC(=O)Cn2ccnn2)OCCC1 52156,c1(C(=O)NCC(Cn2cc(NC(=O)CC#N)nn2)OC)cc(C(C)C)ccc1F 52157,Cc1nc(C(=O)Nc2ccnc(-c3ccnc(F)c3Cl)c2)ccc1F 52158,c1(CC)ccc(C(=O)NCCC(C)NC(=O)CCC2CCC(=O)NC2)cc1 52159,C1(NC(c2c(CC)nc(C)[nH]2)=O)CCN(C(C2CCN(C(N)=O)CC2)=O)CC1C 52160,c1(CC)cccc(C(N2CCOCC2CCNC(c2ncccc2F)=O)=O)c1N 52161,C1(C(N(CCC(C)NC(C=Cc2scc(C)n2)=O)C)=O)CCCCN1N=O 52162,C12(C(=O)NCCN(CCC)C(C3(C)CC(C(F)(F)F)C3)=O)CCCCC1OCC2 52163,C12(NC(=O)Cc3cnns3)CC(CNC(C3CC3c3cccs3)=O)(C1)C2 52164,O=S(=O)(c1ccc(Br)cc1N1CCC(NC2CCOCC2)CC1)N1CC2CC1C2 52165,C(=O)(C1=C(C)CCCC1(C)C)NCCC(CNC(c1cc(C)oc1)=O)O 52166,c1(C(=O)NCCN(C(COCC)=O)CC(C)O)sc2c(Br)csc2c1C 52167,c1(CCNC(C(C)N(C(C(n2ncc(C)c2)C)=O)C2CC2)=O)ccc(C)nc1 52168,CC1=NOC(C)(CNC(=O)CCc2ccncc2Br)C1.n12cc(nn1)C2(C)C 52169,c1(SC)ncc(CN2CCC(NC(c3ccc(-c4ccccc4)s3)=O)C2)c(Cl)n1 52170,C1(C(N(C(C(C)SC)C)C)=O)CC2(CCC2)CN1C(=O)C(Cl)Cl 52171,c1(C(=O)NCC(C)(C)OCCNC(C2C(C)CCOC2)=O)cnn2c1CCC2 52172,Cc1cc(C(=O)NC2CC(NC(c3cc(Cl)ncc3Cl)=O)C2)cc(C)c1Br 52173,C1(C(N(CCCN2CCCC2)C)=O)CCN(C(=O)C2CC(N=[N+]=[N-])C2)O1 52174,N1(C(c2cncc(C)n2)=O)CCCC2(C1)CN(C(c1cccc3nscc13)=O)C2 52175,C1(c2n(C)cnn2)CCCN(C(=O)CN2C(=O)CC2=O)C1 52176,CC1(C)CCCC(CN=c2[nH]nco2)C1.C(=O)(C(C)(C)C(N)=O)N 52177,Cc1cc(C(N2CC3CC3C2C(N2CC3C(CO)C3C2)=O)=O)ncn1 52178,c1(C(C)C)cccc(C(N2CC(NC(C3CC4CCC4C3)=O)C(C)C2)=O)n1 52179,n1(C(C)C)cnc2ccc(CNc3ccc(-n4ccnc4)cc3)cc12 52180,c1(NC(C2N(Cc3cccc(C(=O)O)c3)CCC2)=O)ccc(I)c(Br)c1 52181,C1(NC(C(C)=C(CC)C)=O)CCCN(C(C2(CCOC)CC2)=O)CC1 52182,Cc1sc(O)nc1C(=O)NC1CCCCC1N(C)C(c1cc(C(F)F)ncn1)=O 52183,C(=O)(C1=CCC(C)(C)CC1)NCCC(C)NC(=O)CCCOc1cccc(F)c1 52184,N1(C(=O)OC(C)(C)C)CCC2(CCC2)C(NC(C2(N=[N+]=[N-])CC2)=O)C1 52185,c1(CNC(C2CCC(CNC(C3CC34CCOC4)=O)O2)=O)cnccc1Cl 52186,Cc1ccnnc1C(N1CCCC1C(C)(C)C(=O)N(C)Cc1ncco1)=O 52187,c1(OC)nc(N2CCC2(C)C(=O)NCCN2CCCCCC2)ncc1Br 52188,N1(C(C2=CCCC2C)=O)CC(CO)C2(C1)CN(C(c1sccc1Cl)=O)C2 52189,C1(C(=O)NCC(C)CN(C)C(c2cccc(N)c2N)=O)CC2CCC(C1)C2 52190,c1(C(=O)NC2CCN(C(C3(C)CCCOC3)=O)C2)cccc(S(C)(=O)=O)c1 52191,CCC(CN=c1cccc(S(=O)(=O)NCCN(C2CC2)CC)[nH]1)N(C)C 52192,Cc1cc(C(=O)NCCNC(=O)CC(F)(F)Br)n(C(C)(C)C)n1 52193,n1(CC)nc(C(=O)NC2CN(C(C3(Br)CC34CCC4)=O)C2)cc1C 52194,c1(OC)nc(C(=O)NC(C)(CNC(=O)CCc2nccs2)C2CC2)sc1C 52195,c1(CNC(CC(=O)NCC#C)=O)nnn(C)c1C(=O)NC(CO)C(C)(C)C 52196,c1(C(=O)NC2CCN(C(c3c(O)cccc3Br)=O)C2)ccc(O)c([N+](=O)[O-])c1 52197,C1(CC(N2CCC(NC(CCOC)=O)C2)=O)CCCC(C)C1 52198,N1(C(=O)Cc2cnsc2)CCC2CN(C(=O)Cc3cccc(F)c3F)CCC2C1 52199,c1(CC)ccc(C(=O)NCC(C)N(C(=O)COCc2ccccc2)C)o1 52200,N1(C(c2ccc(CSCC)cc2)=O)CCC(O)C(NC(=O)CC(C)C(F)F)C1 52201,N1(C(C2C(CC)C2)=O)CCC2(CC1)CC(NC(c1cnc(C(C)(C)C)s1)=O)CO2 52202,C12(C(N(CCCNC(=O)CC(F)(F)F)CC)=O)CCCC(CCC1)C2 52203,C1(C(=O)NCC(=O)OCC)(CC)CCCN(C(C2CC3CCCC3C2)=O)C1 52204,C(=O)(CCCCC(N)=O)NCCOc1ccc(OC)cc1.C12CCCCN1C2 52205,n1(CCc2n(CC)nc(-c3ccnc(Cl)c3)n2)cc(Br)ccc1=O 52206,C1(C(=O)NC2(CC)CN(C(C3C4(CC4)C34CC4)=O)C2)CCC2CC1C2(C)C 52207,CC1(C)COC(CCC(=O)NCCC2(O)CN(C(c3cc(O)cs3)=O)C2)C1 52208,c1(C(=O)NC)cccc(OCC(=O)NC2CCCC2NC(C2(C)CC2C)=O)c1 52209,C1(Cc2n(-c3cnc(C)s3)nc(-c3cccs3)n2)CCC(C)(C)CC1 52210,N1(C(C=CCOC)=O)CCOCC1CC1CCN(C(C2CC2C(F)(F)F)=O)CC1 52211,N1(CC(=O)NC2CN(C(CCCCC#C)=O)CC2O)C(=O)NC(C)(CC)C1=O 52212,c1(OCC)ncccc1C(=O)NC1CCCCC1NC(C12CCCC1(CF)C2)=O 52213,N1(C(C)=O)CC(O)CC1C(N1CCSCC1CCNC(=O)CC(=O)N(C)C)=O 52214,C1(C(=O)NC(C)CN2CCOCC2)CCOCCN1C(C1CC1(C)C(=O)OC)=O 52215,C1(NC(C2(C)CCCC2)c2nnnn2C2(C)CC2)CC12CCCCC2 52216,N1(CC(C)CC(F)F)CC(=O)N(CCSCCn2ccnc2)C1=O 52217,CCCC(O)C(=O)NC1CN(C(c2ncncc2Br)=O)CC1C 52218,N1(C(c2c(CCC)n(CC)nn2)=O)CC2(NC(c3ccc(C)n3C)=O)CCC1C2 52219,N1(C(CCCCCC)=O)CCC(CNC(c2cccc(C)c2F)=O)C(F)(F)C1 52220,Cc1cc(CCC(=O)NC2CCN(C(=O)CNC(=O)C(C)C)CC2F)ccc1O 52221,C(=O)(C(C)(C)C(=O)NCc1c(Br)nnn1C)N(C)C 52222,CCCCC(CN=c1[nH]cnc(Cl)c1[N+](=O)[O-])NC(=O)C1CCc2ccccc21 52223,C(=O)(C(C)(O)CC(C)C)NCC(CO)NC(c1ccc(OCCC)cc1C)=O 52224,CCCCCCC(=O)NC1CC2(C1)CC(CNC(C1CC3C(C1)C3(C)C)=O)C2 52225,C1(C(NOC(C)C)=O)CN(C(C2CC(C)(C)CN2C)=O)CCN1C 52226,C1(=O)CC(C)CC(=O)NC2CN1CCC2C(F)(F)F.C1(OCC)CC1C(=O)NC 52227,c1(C(=O)NCC2CCN(C(C(C)CF)=O)C2)cnnc2ccccc12 52228,N1(C(C2CC(C#C)(O)C2)=O)CC2CC(NC(=O)C(C)OCC(C)C)CC1C2 52229,Cc1ccc(N)cc1C(N1CC2(NC(=O)C(CO)NC(N)=O)CC1C2)=O 52230,N1(C(C(C2CCC2)OCC)=O)CCN(C(c2cccc(N)c2F)=O)CCC1C 52231,CCC(C)CC(=O)C(=O)N(CC(=O)NCCc1ccc(F)cc1)CC 52232,C(CC(C(=O)NC(=O)NCc1ccccc1)N1CCCC1SC)SC.C(C)(C)(C)O 52233,Cc1cccc2oc(C(=O)NC3CC(O)CN(C(c4ncc[nH]c4=O)=O)C3)cc12 52234,CC1(C(=O)NC2CCCN(C(=O)C3CC3)C2)CCCN(Cc2cccc(CO)c2)C1 52235,c1(C(=O)NCc2occ(C(N(C)CC3C(C)OCC3)=O)n2)cc2ccccn2c1 52236,c1(C(C(=O)NCc2nncs2)NC(CSC(C)C)=O)cnn(C)c1 52237,CN1CC2CC1CN2C(C1CC(NC(c2ncn3c2CCC3)=O)C1(C)C)=O 52238,c1(NC(CC(=O)Nc2cccc(OC)c2C)C)ccc2c[nH]nc2c1 52239,C(=O)(C(O)CC(=O)OC(C)(C)C)NCCC(C)(C)NC(c1cnc[nH]1)=O 52240,C(c1cnccn1)=CC(=O)NC1CCCC1CNC(C1CCCCC1O)=O 52241,N1(C(C2CCC(C)(CC)O2)=O)CCN(C(c2cc(SC)oc2C)=O)C2COCC12 52242,N1(C(C(=O)NC(C(C)C)(C)Cc2ccccc2)=O)CCNCCC1C 52243,N1(C(CC=CC=C)=O)CCC(C)(C)C(C(=O)NC(C2(OC)CCC2)C)C1 52244,C1(NC(c2c(OC)cccn2)=O)CCN(C(=O)C(O)Cc2[nH]cnc2C)CC1F 52245,Cc1cc2nc(N3CCC(NC(=O)C(F)(F)c4cscn4)CC3C)cc(=O)n2o1 52246,c1(C(=O)NC(CNC(CC(=C)C)=O)(C)CC)ccc(-c2cnco2)cc1 52247,C1(NC(CCOCC(C)C)=O)CCCC1C(=O)NOCC(C)(C)O 52248,N1(C(C2CC(CC)(CC)C2)=O)CCC(NC(C2CCC(=O)C2)=O)C(F)(F)CC1 52249,Cn1c(I)cc2c(N(C(=O)CC(F)(F)F)C3CCNC3)ncnc12 52250,N1(C(C(CC)Br)=O)CCC2C(C1)OCCN2C(C1=NC(=O)N1C)=O 52251,C=CC1CN(C(=O)CCN(C)CC)CC1NC(C1CCN(C2CCCCC2)C1)=O 52252,c1(C(=O)NCC(C)NC(c2cn(CC)nc2C(C)(C)C)=O)coc2ccccc12 52253,c1(C(=O)NCCCN(C(C(CC=CC)C)=O)C)cc(OC)cc2ccoc12 52254,CC(C)(CC(=O)NC1CC(n2cncn2)C1)NC(C1CC2CC2C1)=O 52255,C1(N(C(C)C)CCN(C)C)COc2cc(Br)ccc2C1 52256,N1(C(c2c(OC)scc2)=O)CCC(NC(=O)CNc2ncccn2)C(CO)C1 52257,C(=O)(C(CC)CC(F)(F)F)NCC(CC=C)NC(C1(CC#C)CCC1)=O 52258,CC(C)(CNC(C1CCC1C#N)=O)CC(=O)N1CCCCC1C1(O)CC1 52259,N1(C(C2(CC)CCN(C(C3CCCN3C=O)=O)C2)=O)CCCCC(CO)C1 52260,C=C1CC2(C1)CC(C(=O)N(C(CNC(c1ncccc1F)=O)C1CC1)C)C2 52261,N1(C(C2C(C)(CC)C2)=O)CC2(CCN2C(=O)CCN(S(C)(=O)=O)C)C1 52262,C1(NC(C(CC=C)CNC(C2(O)CCC2)=O)=O)C2CCN(CC2)C1C 52263,C1(NC(C(n2cc(CNC(COCCCC)=O)nn2)C)=O)CN(CC)C(=O)O1 52264,N1(C(Cc2n(C)ccn2)=O)CC=C(C(=O)NCc2ccc(F)c(F)c2)CC1 52265,CN1CCC(C(=O)NC2CS(=O)(=O)CC2NC(C23CC(C2)C3)=O)c2ccccc21 52266,c1(C(=O)NCC2C(NC(c3c(N)c(F)ccc3)=O)C2)cccc2c1OC(F)(F)O2 52267,C(=O)(CC1=NNC(=O)C1)NCCOCCCNC(C1C(C(C)C)CCC1)=O 52268,C1(C(NOC)=O)CCCN(c2ccc(C)nn2)C1 52269,C1(c2onc(C)n2)CCCCN1C(c1ncnn1C)C(=O)NC1(C)CC1 52270,c1(C(N2CC3C(NC(C4N(CC)CCC4)=O)C3C2)=O)cc(OC)cc2c1CCC2 52271,c1(C(=O)NC(C(C)C)CNC(c2coc(CO)c2)=O)cc(Cl)cn1C 52272,Cc1cccc(C(N2CCCC(CNc3nccnc3C#N)C2)=O)c1Cl 52273,C1(CCCNC(CCCOC(C)C)=O)CCN(C(=O)CC2CCOC2)CC1 52274,CCC(C)CC(C)N(C(=O)CN(C(=O)CNC(C1(OC)CC1)=O)C(C)C)C 52275,c1(OC)ccc(C)c(CN2CCC3(CC3C(=O)NCC=Cc3ccccc3)C2)c1 52276,N1(C(CC=C)=O)CC2CC(C)N(C(=O)CCOc3ccc(Cl)cc3)C2C1 52277,c1(OC(C)C(=O)N(CC(C)NC(C2(CN(C)C(C)C)CC2)=O)C)cccnc1 52278,c1(C(=O)NC2C(NC(C3(CC)CCNC3=O)=O)CCCC2)cnc(Cl)cc1N 52279,C12(CNC(Cc3ncc(C)o3)=O)CC1CN(C(=O)C=Cc1cnc[nH]1)C2 52280,CCCCC(C)CCC(=O)NC(Cc1cnn(C)c1O)C(=O)NCCCN=[N+]=[N-] 52281,c1(Cc2nc(N(C)C)sc2)nc(-c2cc(Cl)c(Cl)s2)n(C2CCS(=O)(=O)C2)n1 52282,c1(SC)c(C(=O)NC2CC2NC(c2cnc(OC(C)C)nc2)=O)cnn1C 52283,C1(C)(NC(C(CNC(CN(C)CC)=O)C)=O)CN2CCC1CC2 52284,N1(C(C(=Cc2cn[nH]c2)C)=O)CC2CCN(C(C3CCCCO3)=O)C2C1 52285,C(=O)(NNC(=O)C1OCCc2ccccc21)NC(CC)C 52286,N(C1COc2c[nH]nc21)C(CCC(CC)NC(c1cccc(F)c1N)=O)=O 52287,CCC(C)C(O)CC(=O)NCC(C)(F)CNC(c1ccnc2cc[nH]c12)=O 52288,O=C(CCCCCCBr)N1CCN(Cc2c(Br)cc(F)cc2Br)CC1C(F)(F)F 52289,C(=O)(N=c1cccn[nH]1)c1c(NC(c2n(C)ncc2Br)=O)ccs1 52290,C(CCC(C)C)(C(=O)NC1CN(C)CC1C)NC(COCCCOC)=O 52291,N1(C(C2(CC#C)CC=CCC2)=O)CCC2(CC1)CN(C(c1nccnc1C)=O)C2 52292,CC(CCC(=O)NCC1COC(C)(C)C1)NC(=O)C(F)C1CCC1 52293,c1(C(C2CCCCC2)NC(c2cn(C)cn2)C)cccc(C(F)(F)F)c1 52294,Cc1ncc(C#N)c(N(C)CC2CN(C(c3c(C)cc(O)cc3O)=O)C2)n1 52295,C(=O)(CS(=O)(=O)C1CC1)NC1CCN(C(C2(CCC)CC(=O)C2)=O)CC1C 52296,C1(C(=O)NCC2(NC(C(C)c3ccon3)=O)CCC2)CSCN1C(=O)C(C)(C)C 52297,N1(C(c2cc(Oc3cc(OC)no3)c(F)cc2)=O)C2CCC(C2)C1CC(=O)OC 52298,C(c1cncn1C)=CC(=O)NC1CC(CNC(CSCCC)=O)C1 52299,Cc1ccc(C(=O)N(CCNC(C2CC(C)CO2)=O)CCOCCO)nc1 52300,n1(CC(=O)NCC2N(C(COCC(=C)C)=O)CCC2C)cccc(C)c1=O 52301,CCC(CN(C)C)CC(=O)NC(C)(CO)C(=O)N(C)CCN(C)CCO 52302,CC1C2CC(C2NC(=O)CSc2cccc[n+]2[O-])N1C(=O)CSC1CCCCO1 52303,C1(CC)CCN(C(C2CN(C(C3(O)CCCC3)=O)CC23CC3)=O)CCO1 52304,C1(C(N2CC(COC)(NC(C3CCCC3F)=O)C2)=O)CC(O)C(F)C1 52305,N1(C(C2(C(=O)O)CC(c3cccc(OC)c3)C2)=O)CCN(C(C)=O)CC1C 52306,N1(C(c2ccc(OCC=C)cc2)C(=O)NC)CCCC(C)(OC)C1 52307,C1(C(=O)NC2CCCC(N(C(=O)C=CBr)C)C2)CC2(CCC2=O)C1 52308,C(=O)(C#CC1CCCCO1)NC1CCCN(C(C)=O)C1C 52309,Cc1[nH]c(C#N)cc1C(=O)NC(C)(CNC(=O)CC(=O)NC1CC1)Cn1cccn1 52310,c1(CC(=O)NC2(CC(=O)N(CCCSCC)C)CCC2)cnn(CC)c1 52311,Cc1ccc(CC(=O)NC(C)C(C)NC(c2ccnn2C2CCC2)=O)cc1 52312,CCC(CC)C(C)C(=O)NC(CO)C(C)NC(c1cccc(C(=O)NC)c1)=O 52313,CC(C)(CCC(=O)N1CCC(=CCNC(=O)CC2CCC(=O)N2)CC1)[N+](=O)[O-] 52314,C1(CN2CCC(C(N)=O)C2)CCC2(CCC3(CC2)OCCO3)O1 52315,C=CC1(C(=O)N(C)Cc2cscn2)CCN(C(c2cc(CCC)on2)=O)C1 52316,N=c1cc(C(=O)NCC2CCCC(NC(=O)C=Cc3cccs3)C2)cc[nH]1 52317,C1(CNC(c2c(CC)c[nH]c2)=O)CCCC(CNC(=O)CCC2CCCCO2)C1 52318,CC(CC(=O)c1cccc(F)c1)C(=O)Nc1ccnc(OCCO)c1 52319,c1(CC)nc(C(N2CCC(C(C)NC(C3(CO)CCOC3)=O)CC2)=O)c(N)s1 52320,c1(SC)cc(C)ccc1C(=O)NCC(C(C)C)NC(=O)C(C)(O)C1CC1 52321,N1(C(CC(C)C)=O)CCC2(CC1)CC2C(=O)Nc1cc(I)ncn1 52322,c1(NC)ccc(C(=O)NC2CC2CNC(c2sc(F)cc2Cl)=O)c(Cl)c1 52323,C1(NC(C2(NC(CCC)=O)CC2(C)C)=O)CCn2ccnc2C1.C1C(=O)N1 52324,C1(F)(C(=O)NC2CN(Cc3c(C)noc3C)CC2(F)F)CCCCC1(F)F 52325,N1(C(CCC=CCC=C)=O)CC(C)CCC1CNC(=O)Cc1cnsc1 52326,C1(NC(c2ccncc2F)=O)CCCC12CN(C(c1sccc1F)=O)C2 52327,CC1CCN(C(C2(O)CC2)=O)C1CNC(c1cnn(C2CC2)c1)=O 52328,N1(C(c2cnc(OC)s2)=O)CC2CC(C)N(C(C3(F)CCCCC3)=O)C2C1 52329,CC1(C(N2CCOC(CNC(=O)CSCc3ccncc3)C2)=O)CC(C#N)C1 52330,C(=O)(C(C)(C)S(C)(=O)=O)NC1CCCC(NC(c2c(NC)ccc(F)c2)=O)C1 52331,C1(C)(CNC(c2cc(OC)n(C)n2)=O)CCCN(C(c2cn(C)nc2OC)=O)C1 52332,C(C(C)(C)CC(=O)NCCC1CCN(C(c2ccc(C3CC3)nc2)=O)C1)N(C)C 52333,c1(N2CCC(N(C(CC)CC)CCn3cc(C)cc3C)CC2)ncccc1C#N 52334,CC(C)CC(CNC(C1(P(C)(C)=O)CC1)=O)NC(C1CCCC(CF)C1)=O 52335,N1(C(c2cc(C)ns2)=O)CC2CC(C1)CN(C(c1ccc(C(O)CF)cc1)=O)C2 52336,c1(C(=O)NC2C=CC(CNC(c3cnns3)=O)C2)ccc(OCCO)cc1 52337,O=C(C(=O)N=c1nc[nH]n1-c1ccccn1)N1CCC(C(O)CO)CC1 52338,n1(CC(=O)Nc2cccc(Cc3nc[nH]n3)c2)cc(C(F)(F)F)c2ccccc12 52339,c1(CNC(C2CCCNC2=O)=O)ccccc1O 52340,C1(C=O)C(C(=O)O)C1(C)C.C(=O)(C(=O)NCC)NC(c1nn[nH]n1)C 52341,c1(C(N2CC(CC(C)NC(C(CCCC#C)C)=O)C2)=O)cc(C)c2occc2c1 52342,CC1CC(C)N(C(=O)CC2CCCCC2)CCN1C(c1nccc(Br)c1O)=O 52343,n1(CC(=O)NC2CC(C)(NC(C(C3CCC3)OCC)=O)C2)nnc2c1CCCC2 52344,N1(C(C2CN(C)C2)=O)CC(NC(=O)Cc2csc(NC=O)n2)C2CCCCC12 52345,C12(C(N3CCC(CNC(CCCC=C)=O)CC3)=O)CC3CC(CC(C3)O1)C2 52346,O=C(C#CC1CCC1)NC1CC(NC(=O)C=CCN2CCCCC2)C12CCC2 52347,C1(CNC(Cc2c(C)nc[nH]2)=O)CCCCCN1C(c1cnn(CC2CC2)c1)=O 52348,c1(CN2C3CN(C(C4C5COCC45)=O)C(C3)C2)cc(F)c(F)c(Cl)c1F 52349,N1(C(c2cc(OC)ncn2)=O)CC2(CCN(C(c3ccc(Cl)nc3Cl)=O)C2)C1 52350,C1(NC(C(C)SC)=O)CCCC1(C)NC(=O)Cn1nnn(-c2cccs2)c1=O 52351,C1(CNCC2CCCC2C(N(C)CC2(CC(C)(C)C)CC2)=O)CC(F)(F)C1 52352,c1(C2OCCN(C(c3cc(Br)cc(Br)c3)=O)C2)cc(F)c(Cl)cc1Cl 52353,CC(C)C(C(=O)NCCCS(N)(=O)=O)NC(=O)Cn1cnnn1 52354,c1(C(N2C(CNC(c3coc(Cl)c3)=O)CC(F)(F)C2)=O)cn2c(n1)CCCC2 52355,C1(NC(C(N(C)O)=O)C2CC2)CCS(=O)(=O)CC1 52356,c1(OC)cc(CO)ccc1C(=O)N(C1CN(C(C23CCCC2C3)=O)CC12CC2)C 52357,N1(C(c2nc(OCC)oc2)=O)CC2(CCC2NC(=O)C(S(C)(=O)=O)C2CC2)C1 52358,CC(CO)C(=O)NCC(C)(F)CNC(c1n[nH]cc1C1CC1)=O 52359,C1(NC(c2c(C)nc(O)s2)=O)(CO)CCCN(C(=O)CC(C)C(C)C)C1 52360,c12ncnc(Cl)c1N2CCO.C1(NC(C)C)CCCN(C(=O)OC(C)(C)C)C1 52361,C(CCC(C)C(C(=O)NCC(C)C)N1CCN(C2CC(CSC)C2)CC1)=C(C)C 52362,c1(OC)ncc(-c2cc(F)ncc2F)cc1C(=O)NCc1nn[nH]n1 52363,CCC(C)(C)CCCC(=O)NC(C)CC(=O)Nc1ccc(F)cc1 52364,N1(C(c2cn(C3CC3)nn2)=O)CCCC(C2CCN(CC3CC3)C2)C1 52365,C(=O)(C1=CC2(CN(C(c3cc(C)sn3)=O)C2)OC1)NCC1(OC)CCOC1 52366,n1(C(C(=O)N(CC(C)NC(c2c(C)oc(C#N)c2)=O)C)C)nc([N+](=O)[O-])cc1C 52367,c1(OC(C)C(N2CCN(C(C3C=CS(=O)(=O)C3)=O)CC2)=O)cccc(F)c1 52368,c1(C(N2CC(CC=C)(NC(C3CCC(C)(C)C3)=O)C2)=O)cnc2sc(C)c(C)n12 52369,C(=O)(C(C)(C)CCC#N)NCCC1CCN(C(c2c(C)nc(Cl)cc2)=O)C1 52370,c1(C(N2CC(NC(C3CC4(C3)CC4F)=O)CC(C)C2)=O)cccc2cccnc12 52371,c1(C(=O)NC2C(NC(c3c(CC)n[nH]c3)=O)COCC2)n[nH]c2c1CCC2 52372,S(=O)(=O)(c1ccc(N2CCN(C(C3CC3C)=O)CC2)nc1)NCCCCC 52373,c1(NC(C2(C)CCN(Cc3c(C)c(F)c(F)cc3)C2)=O)cc2[nH]ccc2cc1Cl 52374,C=CC1CN(C(c2c(C)nn(C)c2C)C(=O)NC2CCC2)CC1O 52375,C#CCCC(O)C(=O)NC1(CO)CCCN(C(c2c[nH]nc2CC)=O)C1 52376,C1(C(N(C2CC(=C)C2)C)=O)CCCC1NC(=O)C(C)CN1CCCC1 52377,c1(C(N2CC(NC(Cc3c(C)non3)=O)C(C)C2)=O)cnc2sccc2c1 52378,N1(C(c2c(C)nn(C)c2C)=O)CCN(C(c2cccc3c2CCC3)=O)CC(O)C1 52379,C1(NC(c2c(C)cns2)=O)CN(C(C2CC(F)C(=O)N2)=O)CC2(CCC2)C1 52380,C(=O)(CCCC(=O)N1CC=CC(NC(=O)C(C)C(C)O)C1)NC 52381,c1(OC)ccnc(NCC(=O)NC2CC2CNC(c2cc(Cl)cs2)=O)n1 52382,N1(N(C)C)CCN(C(c2ccnc(CSc3nc(C(C)OC)sc3)c2)=O)CC1 52383,C1(C)(C(=O)NCC(C2(O)CCN(C(C(C)OC(C)=O)=O)C2)C)CCCN(C)C1 52384,N1(C(CC(CN(C)C)O)=O)CC=C(CC(=O)N2CCCC(N(C)C)CC2)CC1 52385,N1(C(c2cncc(C#C)c2)=O)CC2CC(NC(=O)C=Cc3cncs3)C(C2)C1 52386,c1(NC(C)=O)ccc(NC(C2CCCN(Cc3ccncc3O)C2)=O)cc1 52387,c1(C(=O)NCCCOCCC(=O)N(C(C)CCO)C)cnn(C)c1 52388,C1(C(=O)NCc2c(C(=O)NC(Cn3ncc(C)c3)C)scc2)CC2CCCC2C1 52389,CCC(C)C(O)C(C)C(=O)N1CCOC(CN(C(=O)CCC(C)C)C)C1 52390,C(=O)(C1Cc2ccc(Cl)cc21)N1CC(CNC(c2cc(F)ccc2O)=O)OCC1 52391,c1(OC)ccc(CC(N2CCC2CNC(C2C(Cl)(Cl)C23CC3)=O)=O)cc1OC 52392,N1(C(C2C(NC(c3c(C)[nH]c(C)c3C)=O)COCC2)=O)CCCC2(CC(O)C2)C1 52393,c1(C(=O)NC2CCCC(N(C(CCC#C)=O)C)C2)c(Cl)ccc([N+](=O)[O-])c1Cl 52394,c1(C(=O)NCCC2N(C(C#CC(C)C)=O)CCCC2C)ccn2ccnc2n1 52395,Cc1ccc(C(N2CC(F)CC2CNC(=O)C(C)NC(=O)C(C)(C)C)=O)nn1 52396,C(=O)(CCCCCC(C)(C)C)NC1CN(C(c2c(C)oc(Cl)n2)=O)CC1F 52397,C1(C(=O)NCc2c(OCC(=C)C)cccc2)CC(F)CN(C(=O)CCN(C)C)C1 52398,C1(C(N2CCC(CC)C2)=O)COCCN(C(C2CC(N=[N+]=[N-])C2)=O)C1 52399,CC1(C)CN(C(C2CC(F)C(=O)N2)=O)CC(C)(C)C1 52400,C#CC1CCCC(NC(C2CCOC2CNC(=O)Cc2c(C)cnn2C)=O)C1 52401,C(=O)(CC1=CCOCC1)NCCNC(=O)CC(F)F 52402,N1(C(C2(CC)CC(OC)C2)=O)CCC(O)(CC(=O)NC2CCCC(O)C2)CC1 52403,N1(C(c2cc(O)ncc2Br)=O)CCC(NC(C2(C3CC3)CCC2)=O)C(O)C1 52404,C=CCC(C)(C)CC(=O)NCc1cc[nH]c1C(=O)NCC1CC2CC1CC2O 52405,C(c1ccccn1)=C(C)C(=O)NCC1(C(C)NC(c2ccnc(C)n2)=O)CC1 52406,C1(C)(CN(C(c2ccc(Br)c(F)c2)C(=O)O)C)CC2(C1)CC(F)(F)C2 52407,C(=O)(C(C(C)C)C(C)C)N1CCOCC(C(N2CCC(C(=O)OCC)C2)=O)C1 52408,C(=O)(C1CCCc2ncc(C)n21)N1CCN(C(C(CCCC=C)(C)C)=O)CC1C 52409,C1(CCNC(CNC(C)=O)=O)CCN(C(c2c[nH]c(=N)nc2C)=O)CCC1(F)F 52410,C(=O)(CC(O)CC(C)C)NC(CCSC)C(=O)NCC1(C)CC(C)C1 52411,N1(C(C(CC)C)=O)CCC2(CCCC2CNC(=O)CCOC2CCCC2)CC1 52412,C1(C(=O)NCC(O)Cc2ccccc2)C2CCC(C2)N1C(c1cccc(F)n1)=O 52413,C(=O)(CCC(O)C(C)(C)C)N1CC(CNC(c2nc(CC)oc2)=O)C(C)CC1 52414,C(=O)(C(O)CCc1ccccc1)NC1C(CNC(=O)C(c2ccccc2)O)COC1 52415,n1(C(C)C(=O)O)cc(C2(O)CN(C(=O)Cc3ccccn3)C2)nn1.C1(=O)C(C)N1 52416,CC1(C)CC(NC(=O)CCc2ccc(F)cc2Cl)CN(C(=O)Cc2nc[nH]n2)C1 52417,c1(C(N2CCC(NC(c3c(C)[nH][nH]c3=N)=O)C2)=O)ccc(C)c2ccccc12 52418,Cc1nc(NCC(C)(C2CC2)NC(c2ccsc2C)=O)c(C)c(O)n1 52419,C1(NC(CNC(C(CC)C)=O)=O)CCN(C(c2c[nH]c(=N)nc2C)=O)C12CC2 52420,n1(CC)ncc(C(=O)NCc2ocnc2C(=O)NC2(C)CCOC2C)c1C 52421,N1(C(C(C)O)=O)CCN(C(C(=O)NCC2CCCO2)c2ccon2)CC1 52422,CCC(C)(C)C(O)C(=O)N1CC(N(C)C(c2ccc(OC)c(F)c2)=O)C(C)(C)C1 52423,c1(C(=O)NC(C)CN(C)C(c2n[nH]cc2F)=O)ccc(CN2CCCC2=O)cc1 52424,C1(NC(C=CSC)=O)C(C)CCN(C(c2cnc(C3CC3)o2)=O)C1C 52425,CC1CCCCC1(C)C(=O)NC1CCCN(C(c2csc(O)n2)=O)C1C 52426,N1(C(c2c(C)ccc(C)c2)=O)CCCCC2(CCN(CCC3CCCO3)C2)C1 52427,N1(C(C(CC(=O)OC)N(C)C)=O)CC2CCC1CN2C(c1coc(N(C)C)n1)=O 52428,N1(C(c2c(CC)ncs2)=O)CCCN(C(c2ccc(O)c(O)c2)=O)CC1C 52429,C1(CNC(c2c[nH]cc2Br)=O)CC2(CCC2)CN1C(=O)C=Cc1ccc(O)cc1 52430,N1(C(C=CC=CC)=O)CCCCC2(C1)CN(C(c1ccc(OCOC)cc1)=O)C2 52431,c1(C(=O)NCc2c(C(N3CC(C#CC)C3)=O)nn(C)c2)cc2ccccn2c1 52432,C1(C)(CNC(C2(C)CC(C)(C)C2)=O)CCCN(C(C2OCC3CCCC23)=O)C1 52433,C1(C(N2CCC(NC(c3c(C)[nH][nH]c3=N)=O)C2C)=O)CCC2(CCC2)O1 52434,C(=O)(C(C(C)(C)C)N1CCNC1=O)NCC(CO)NC(c1cc(C)on1)=O 52435,c1(C(=O)Nc2scc(CN(C)C)n2)ccc2cc(I)cnc2c1 52436,Cc1cc(C(=O)NC(C(=O)N(C)Cc2nc[nH]n2)C2CCCC2)ncc1N 52437,N1(C(C2(C)CCCN2C(c2cnn3ccncc23)=O)=O)CCn2cccc2C1 52438,CCCCC(CC)Nc1nccc(N2CCN(C(=O)CCNC(C)C)CC2)n1 52439,C=CCCCCCCCCc1nc(CCCCC)nn1C1CCC1 52440,CCCC(C(=O)NCC(F)CNC(c1ccccc1Cl)=O)NC(N)=O 52441,Cc1ncnc(C)c1CC(=O)NC1CC2CN(C(=O)C(C)n3ccnc3)CC12 52442,C=CC(CC)CC(=O)N1CC2CC2(CNC(=O)CN(C)Cc2ccc(C)cc2)C1 52443,CC1(C)NC(=O)CCC1NC(C1CC(NC(=O)C=Cc2ccco2)C1)=O 52444,CCCC(CC)CCC(=O)NCc1cc(C(=O)NC2(c3noc(C)n3)CC2)cs1 52445,CC1CN(C)CC(C(=O)NC2CCC(CCC(=O)NCC(C)(F)F)C2)O1 52446,n1(CC(=O)NC(C)C(C)NC(=O)Cc2cccc(F)c2)nnc2c1CCCC2 52447,O=C(C1=CCS(=O)(=O)C1)N1CC2CC1CN(C(=O)CSc1cccc[n+]1[O-])C2 52448,C12(C(N(CCCNC(C(C(C)(C)C)SC)=O)C)=O)CCC(C)(C(=O)O1)C2(C)C 52449,C(C1CCc2nccn21)NC(C1=NOC(CNC(C(CC)OC)=O)C1)=O 52450,c1(SC)ccccc1C(=O)NC1CN(C(=O)COc2ccsc2Cl)CC1F 52451,C1(C(=O)CNC(C(C)OC2CCCC2)=O)CCC(ON)CC1.C1COCCO1 52452,C1(NC(CC2C(C)OCC2)=O)CC(NC(C2(CC(C)(C)C)CC2)=O)C1(C)C 52453,Cn1ncc2cccc(-c3nc(C4CCOC4)nn3-c3ccnc(O)c3)c12 52454,N1(C(CC(C)(C)C#N)=O)C(CNC(C2(C)CCC(F)(F)C2)=O)CC2CCCCC12 52455,N1(CC(=O)NCC(CN(C(=O)C(C)C2CCCC2)CC)(C)C)CC(=O)N(C)C1=O 52456,c1(CNC2CC(CC(=O)Nc3cnc4cnccn34)C2)c[nH]c2nccc(Cl)c12 52457,C1(CCNC(c2cn(C(C)C)nc2)=O)CCCN(C(=O)Cc2ccsc2)CC1 52458,c1(CC(N2CCCC(NC(C(CC)(C)C)=O)C2)=O)ccc2c(c1)CCCC2 52459,CCCCC(O)C(=O)NC(C1CCCC1)CNC(c1ncc(F)cn1)=O 52460,Cc1cnc2cc(C(=O)NC3CC4CCC3(NC(=O)CNC(N)=O)C4)nn2c1 52461,CCC(CC1CCCC1)C(=O)NC1CCOC(CNC(=O)C=C2CCCCC2)C1 52462,N1(C(C2CCC(C)NC2=O)=O)CCC2(CCN(C(=O)C=Cc3ccsc3)CC2)C1 52463,C(CCCC(=O)NCC(C)N(C(=O)Cn1nnc(-c2cccs2)n1)C)OCC 52464,N1(C(=O)NCC(C2CCCC2)(C)C)CCC(Cn2cncn2)C1 52465,c1(CSCC(=O)NCCN(C(=O)Cn2cccn2)CC)ccc(S(C)(=O)=O)cc1 52466,N1(C(CN(C(=O)Cc2ccc(C#N)cc2)C(C)C)=O)CCS(=O)C(C)C1 52467,c1(OCC=C)ccc(C(=O)NC2(Cc3nc(C(C)(C)C)co3)CNC2)cc1 52468,C1(NC(Cc2ccc(C(=O)NC)cc2)=O)CCN(C(=O)CCNC(C)=O)C(C)C1 52469,c1(NC(c2nnc3ccccn23)CC)nccc(=NC2CCN(CC3CC3)C2)[nH]1 52470,C1(CC(=O)N(C2C(C)CC2)C)CN(C(=O)C(C2CCOCC2)O)CCO1 52471,N1(C(CCC2CCN(C(C(C)CO)=O)CC2)=O)CCCCCC1CO 52472,c1(C(C)C)ccc(C#N)c(NCC2CCCN2C(C2CCCC3CCCN23)=O)n1 52473,c1(C(N2CC(CCNC(C3C(OCC)C3)=O)OCC2)=O)cnc2c(n1)CCCC2 52474,c1(C(=O)NCC2(CNC(Cn3ccc(C)n3)=O)CC2)c(C)cc(Cl)cc1C 52475,Cc1ccccc1CCC(=O)NCCCCCNC(C1CCC(F)C1)=O 52476,c1(C(=O)NCCC(Cc2ccccc2)NC(=O)CC2CC(F)C2)cccc[n+]1[O-] 52477,N1(C(c2nc(CC)sc2)=O)CC(NC(=O)C(C)CCN(C)C)C(C)(C)C1 52478,c1(CC)ccc(C(=O)NCC2CCN2C(=O)CC(=O)OC(C)(C)C)cc1[N+](=O)[O-] 52479,c1(C(=O)NC2CC(C)(CNC(C3(C=C)CC3)=O)C2)c(C)nc2sccn12 52480,c1(C(N(CC(CNC(COCCC=C)=O)C)C)=O)cnc(Cl)s1 52481,c1(C(N2CC(NC(=O)Cn3ccnc3)C(O)C2)=O)ccc(Cl)c2ccccc12 52482,C(=O)(CCCC(C)NC(=O)CC(C)(C)OC)N1CC(CC)SCC1 52483,C(=O)(C(O)CCCNC(=O)CCCC1CC1C)N(CCC(=O)NC)CC 52484,C(=O)(C(C#N)C(C)C)NCCCCNC(C(C(C)C)SC)=O 52485,CC1(C)CCCN(C(=O)C=Cc2cnc(O)nc2O)C1CNC(C1OCCO1)=O 52486,c1(C(CCC)NCC(CC)CCO)cc(OC)c(OC)c(Cl)c1 52487,n1(CC)nc(C)cc1C(=O)NC(C(=O)NCC(F)C1CCC1)C1(O)CCC1 52488,c1(C(N2CC3C(NC(C4(C)CN(C)C(=O)C4)=O)C(C3)C2)=O)cc2c([nH]1)CCCC2 52489,C12(C(=O)NCC3(NC(CNC(N)=O)=O)CCCCCC3)CCCCC1C2(F)F 52490,c1(C(CN2CCC(NC(=O)NCc3n(C)ccn3)CC2)=O)c(Cl)cccc1Cl 52491,C=C(C)c1cccc(NC(=O)C(COCC)NC(=O)CC(C)F)c1 52492,C1(C(=O)OC(C)(C)C)CC2CCC1(CC(=O)O)C2.C12CC(C1)CCC(=O)N2 52493,C1(CC(N2CC(N(C)C(c3ccncn3)=O)C2)=O)NC(=O)CN(C)C1=O 52494,N1(C(CCCOCC=C)C(=O)NCCC)CCC(F)(F)C2(CCOC2)C1 52495,C1(CC)CN(C(=O)CC(F)(F)CC)CCN1C(=O)COc1cc(F)ccc1F 52496,C1(CC)CC(O)CCN1C(C1CCOC1CNC(c1cnnn1C)=O)=O 52497,CCC(CC)C(=O)NCc1csc(C(=O)NC(C)CS(C)=O)c1 52498,c1(SCC(=O)NCC(F)CNC(=O)CCN2CCOC2=O)ccccn1 52499,C1(NC(C=C(C)C)=O)CCC(C)N(C(C2C3COCC23)=O)C1 52500,C=C(C)C1OCCC1CNC(=O)CC1CC(C(=O)OCC)C1 52501,C1(C(CNC(C2C(CC)C2)=O)(C)O)CCN(C(=O)CN(C2CCC2)C)CC1 52502,Cc1ccn2c(C(N3CCOC(CCNC(c4ccccn4)=O)C3)=O)cnc2c1 52503,C1(C(=O)NC2CCCN(C(C3(CC)CC(F)(F)C3)=O)CC2)CC2CCC1C21CC1 52504,C1(CNC(C2CCS2(=O)=O)=O)CCN(C(c2csc(C(F)(F)F)c2)=O)C1 52505,c1(C(N2CC(C)C(CNC(c3cc4c[nH]nc4s3)=O)C2)=O)cc(N)c(Cl)c(O)n1 52506,C(=O)(C1=NOC(C)(C)C1)N(C1CCCC(NC(c2c(CC)[nH]cc2)=O)C1)C 52507,c1(CNC(c2c(C)c[nH]n2)=O)cccc(C(=O)NC(C)CN2CCCC2=O)n1 52508,C#Cc1cccc(CNC(=O)COC2(C)CN(C(C3CCC(=O)C3)=O)C2)c1 52509,c1(C(=O)NCC(CC)NC(=O)C(F)(F)c2csc(Cl)c2)n[nH]c2c1CC(C)CC2 52510,S(=O)(=O)(c1cccc(NC(=O)COCCOC(C)C)c1)NC 52511,C#CCCCC(C)C(=O)NC1CC(C(=O)NCCCN2CCCC2)C1 52512,Cc1cc(C(N2CC(O)(CCNC(C34CCCCC3C4)=O)C2)=O)cc2nc[nH]c12 52513,C1(C(=O)NCC2COC3CC2C3)CCC2(CCOCC2)C1 52514,c1(C(=O)NC2(CCNC(C3CCC(C)C3)=O)CCC2)nc(N(C)C)nc(=N)[nH]1 52515,C(=O)(C(C1CCCC1)NC(=O)CSC)N(C(C)CNC(C)=O)CC 52516,N1(CC(=O)NC(C(C)C)CNC(c2cc(Cl)n[nH]2)=O)CCC(=O)NC1=O 52517,C1(N(C(C(F)=CCC)=O)CC)CCCN(C(c2ccn(CC)n2)=O)C1 52518,n1(C(C)(C)C)ncc(C(N(C2CC2)Cc2ccc(SC3CCC3)nc2)=O)c1Cl 52519,O=S(=O)(c1ccc(Cl)cn1)NC1CCN(Cc2cccc(Br)c2F)C1 52520,C(=O)(CC(CNC(=O)CN(C1CC1)CC)C1CCC1)N(C1CCCCC1)CCC 52521,CC1CC(NC(=O)C(C)(F)F)CCN1C(C1CC(c2ccccc2)O1)=O 52522,c1(C(=O)NC2CCCC2NC(C2(C3CC3)CC=CC2)=O)ccc2nc(O)sc2c1 52523,c1(CN2CC(CNC(C(CC)C)=O)OCC2)nc2ccccc2[nH]1 52524,N1(C(C#CC(C)C)=O)CCCC(C2CC2NC(=O)CC2CCCCCC2)C1 52525,c1(N(CCNC(C=CCCC)=O)C)c(O)nc(=O)n(Cc2ccccc2)c1N 52526,n1(CC(=O)OC)cnc(C)c1C(=O)NC1CC(C)(NC(c2cccnc2C)=O)C1 52527,c1(C(c2n(CC(=C)C)nnn2)NCC2CCO2)c(Cl)ncn1C 52528,O=S(=O)(c1[nH]cc2c1CCS2(=O)=O)Nc1ccncc1C(F)(F)F 52529,Cc1ccnc(NCC2CCCN2C(=O)C(C)Oc2ccccn2)c1[N+](=O)[O-] 52530,C12(N(C)C(C3CCCC3CNC3COCCO3)=O)CCC(CC1)CC2 52531,c1(OCC)ncc(NC(=O)CCCN(c2ccccc2)C(C)=O)cn1 52532,C1(F)(C(=O)NCC2C3CN(C(C4(CC)CCOC4)=O)CC32)CC2(CCC2)C1 52533,C(=O)(C(CCOC)NC(=O)CCc1nc(C)no1)NC(C=C)C1CCC1 52534,N1(C(C2CN(Cc3ccncc3)CC(F)(F)C2)=O)CCN2CC(O)CC2C1 52535,CC1CC(C(=O)Nc2nnc(-c3ccco3)o2)N(C(C2CCCS2)=O)C1 52536,N1(C(C2(C)CC2Br)=O)CCC2(CCCCN(C(c3ccc4cnnn4c3)=O)C2)C1 52537,c1(C(=O)NCCOCCNC(C(C)OCCC=C)=O)cc(Cl)c(Cl)[nH]1 52538,C(=O)(C(F)(F)C(F)(F)F)NC1CCCN(C(c2ccc(OC)s2)=O)CC1 52539,C(=O)(CCCCCCS(N)(=O)=O)N1CCCC(C(N2CC(C)NC(=O)C2)=O)C1 52540,c1(N2CC3(C(NC(C4CC5C=CC4C5)=O)CCC3)C2)c(Cl)cc([N+](=O)[O-])cc1Cl 52541,Cc1cc(C(=O)NCCCOCCNC(=O)C(O)CC(F)F)nc(O)c1 52542,C#CC1(C(=O)NCc2cc(C)c(C(=O)NC(C)C(C)C)o2)CCCC1 52543,C1(C(=O)OCCc2nn(C)cc2C)(COC)COS(=O)(=O)C1 52544,C=CCCC(C(=O)N1CCC(C(F)F)C1)NC(c1ccc(C)cc1)=O 52545,CN1CC=C(c2ccc(CNC(c3ccc(OCCCl)cc3)=O)cn2)CC1 52546,C1(CNC(C2(CC)CCCO2)=O)CC(OC)CN1C(=O)CC1(CN2CCCC2)CC1 52547,c1(C(N(CC(C)(C)C(=O)NC(C2CCCO2)CO)C)=O)cccc2[nH]ccc12 52548,c1(CC(=O)NCC2C=CC(NC(C3CNC(=O)N3)=O)C2)cccc(C(F)(F)F)n1 52549,C1(C(=O)NCC(C)NC(=O)C(C2CC(F)(F)C2)O)CCCN(C)C1 52550,CN1C(=O)CSC1=CC(=O)NC1CC(CNC(c2c(N)cccc2Cl)=O)C1 52551,N1(C(CCC=CC(C)C)=O)CCC(C2CCN(C(c3c[nH]nc3C(F)F)=O)C2)C1 52552,C(=O)(C(F)(F)CN1CCCC1)NCCCN(C)C(C1(F)CCCCC1)=O 52553,c1(C(=O)NC2CCC(C)N(C(=O)CN(C3CCSC3)C)C2)ccc2cnoc2c1 52554,N1(C(c2n(CCC)ccc2)=O)CCCN(C(c2cccnc2)=O)C(C)C1 52555,Cc1c(CNC(C)CCSC)c[nH]c1-c1nn[nH]n1.c12ccc(cc1)CN2 52556,C1(C(C)(CO)NC(c2nc(Cl)cs2)=O)CCN(C(C2CCCCS2)=O)CC1 52557,C1(C(=O)NC(c2ncc[nH]2)CC)(NC(=O)CC2(C)CCCC2)CC(CO)C1 52558,c1(C(=O)NCC(C)CNC(=O)CC(c2ccc(Cl)cc2)O)ccc2c(c1)OCC2 52559,C(=O)(C(CCF)NC(=O)CC(=O)NC1CC1)NC(C)CCCO 52560,C(CS(=O)(=O)CCCCc1ccc(C#N)cc1)N(C)C 52561,N1(C(C2CC(CC)C2)=O)CC2(C(=O)NCC3CC(C(C)(C)C)C3)CC1CCO2 52562,C(=O)(C1=CCCCCC1)NCC(CC=C)NC(C1CC(Cl)(Cl)C1)=O 52563,C1(O)(CNC(c2cc(C)c(F)cc2)=O)CCCN(C(C2C=CCS2)=O)CC1 52564,C1(NC(C=CCCC)=O)CC2(CNC(=O)CC(C)c3cccnc3)CC1CO2 52565,n1(CC)cnc(C(=O)NC(C)C(C2CCCCC2)NC(C2CC(C)(F)C2)=O)n1 52566,N1(C(C2CC(=C3CC3)C2)=O)CCN(C(C2(C3CCC3)CC2)=O)C2COCC12 52567,c1(C(C)C)c[nH][nH]c1=NC(=O)C1CN(C(c2cccc(O)n2)=O)CCC1O 52568,N1(C(C2CCN(C(C)=O)CC2)=O)CCC2(CCCN2C(=O)Cn2cc(C)cn2)C1 52569,Cc1cccc2[nH]cc(CCC(=O)N(C)CCN(C)C(C3CCC34CCC4)=O)c12 52570,c1(NC(CN2C(CCNC3CCN(C)CC3)CC2)=O)cnc2c(n1)CCCC2 52571,N1(C(Cc2c(C)n[nH]c2)=O)CC(NC(=O)C(C)(C)C#N)C(c2ccc(F)cc2)C1 52572,CCCCC(=O)C(=O)NC(CN(C)C)C(=O)N(CC)Cc1ccoc1 52573,C1(N(C)C)CCCN(CC(N2CCC(CNC(C3(OC)CCC3)=O)C2)=O)C1 52574,N1(C(c2cc(N)c(F)c(F)c2Cl)=O)C2CCCC1CN(C(c1ccsc1)=O)C2 52575,C1(CNC(C(C)O)=O)CCCCN(C(=O)CC2CCCC2)CC1 52576,CCC1(CNC(CCc2ccccc2)C(F)F)OCCc2ccccc21 52577,N1(C(COCC)=O)CC(C)(C)CC1CNC(=O)CC1CC(F)(F)C1 52578,c1(C(=O)OCC(CCC(C)=O)(C)C)n[nH]c2c1CC(C)CC2 52579,CCC(O)C(C)C(=O)N1CCCC(CCNC(c2cc(C3CC3)n(C)n2)=O)C1 52580,c1(C(N2CCCCC(CNC(CC3CN(C)C3)=O)C2)=O)cnn2c(=N)[nH]cnc12 52581,N1(C(C(CC)C(C)C)=O)CC2(C1)SCCC2NC(c1cccn2cncc12)=O 52582,C1(C(=O)NCC(c2ccccc2)C)CC(O)CN1C(=O)CC1CC(=O)NC1=O 52583,C#Cc1cc(C(=O)NCCC(O)C(=O)NC(C)CC(=O)NC(C)C)ccc1C 52584,C1(C2CCCCO2)(C(=O)NCC(C)CN(C)C(c2ccc(CO)o2)=O)CCCO1 52585,n1(CC(=O)NCC2(CNC(CCSC)=O)CCC2)cc2ccccc2n1 52586,N1(C(COCCOC)=O)CCC(NC(C2Cc3nccn3C2)=O)C(CO)C1 52587,C1(C(N2CCCC(N(C(CCN3CCN(C)CC3)=O)C)C2)=O)CC(C2CC2)=NO1 52588,CC1CN(CC(=O)CC2CCCNC2=O)C(C)CN1Cc1ccccc1 52589,C1(NC(C2CC(C)(O)C2)=O)CN(C(=O)CC2CCCS2(=O)=O)CCC12CCC2 52590,c12ccc(nc1)C(=O)NC1CCC(C1)N(C)C2.c1(OCC)ccc(C(=O)OC)o1 52591,c1(C(=O)NCC2CCN(C(CCOCCOC)=O)C2)nc(C)c(C)nc1C 52592,N1(C(=O)C=CC2CCCC2)CCC2OCCN(C(C3CCCS3(=O)=O)=O)C2C1 52593,c1(C(N2CC(O)CC(NC(C3CC(CC)C3)=O)C2)=O)n[nH]c2c(C)cccc12 52594,C1(C(C)NC(=O)C=CC2(C)COC2)CCN(C(C2CC2(F)F)=O)CC1 52595,c1(CCC(=O)NC(C(C)NC(C(F)=CC)=O)C)nc(C)cs1 52596,CCC(C)C(C(=O)NC1C2CC3C1C3C2C(=O)NCCCO)OC 52597,C1(CN(C(COCC=C)=O)C)C2CN(C(=O)CCCc3nc(C)no3)CC12 52598,c1(OC(C)C(=O)O)ccc(F)cc1NC(=O)Cc1cc(=O)n(-c2ccccn2)[nH]1 52599,N1(CC)CCC(C(=O)NC23CC(C(=O)NCC(O)C(F)F)(C2)C3)C1 52600,CCC(C)C(C)C(=O)NC1CN(C(=O)C=C(C)Cl)C1 52601,C(=O)(C(CC1CC1)NC(c1ccoc1C(C)C)=O)N1CC(C(N(C)C)=O)C1 52602,N1(C(c2cc(C)sc2C)=O)CC(CNC(=O)C(O)C2CC2)CC(C)(C)C1 52603,N1(C(C2C(C)CC=CC2)=O)CCOCCC1C(=O)N(C1CCC(F)(F)C1)C 52604,N1(C(C(C)N(C(c2cnnn2C)=O)CC)=O)CCN2C(=O)NCC2C1 52605,C1(OCC(=O)NCCC(C)(C)NC(c2cc(C)c(Cl)s2)=O)C#CCCCCC1 52606,CC(=O)C(C)(C)CC(=O)N1CC2(CC(C(=O)NCC3(C)CC3)CO2)C1 52607,N1(C(=O)NCC(N2CCCCC2C)C)CCC2(CCCCC2)CC1 52608,C1(NC(=O)C(N2CCSC3CCC23)=O)(Cn2cnnc2)CC2(CCC2)C1 52609,CC1(CC(=O)NC(CO)C(F)(F)F)CCN(C(c2nccnc2N)=O)C1 52610,CCC(C)CC(C(=O)NCC(C)(C)C(F)(F)F)NC(=O)CN(C)CC 52611,C1(C(=O)NCCC2(OC)CN(C(c3ccnnc3O)=O)C2)CCC(C)NC1=O 52612,C1(=CCNC(C(C)(O)C2CCOCC2)=O)CCN(C(=O)C(F)OC(F)(F)F)CC1 52613,C1(NC(c2cnc(C(F)F)nc2)=O)CC2CC(C1)N(C(c1cnco1)=O)C2 52614,CCC(F)(F)CC(=O)NC(CC1CC1)CC(=O)Nc1cnn(C(C)(C)C)c1 52615,C1(Nc2nccc(=NCc3[nH]nc(CSC)n3)[nH]2)CN(C)C2(CCCC2)C1 52616,c1(CC(=O)N(C(CNC(CC(=C)Br)=O)C)CC)nc(C2CC2)nn1C 52617,c1(C(n2ccnc2)CNC(=O)NC2CCCSC2)cccc(Br)c1Br 52618,c1(C(=O)NC2C3CN(C(C(C(C)C)NC=O)=O)CC32)cc2cc(Cl)ccn2n1 52619,C(=O)(C1=NOC2(CCC2)C1)N1CCC(C(N(CCOC)CC)=O)(CO)C1 52620,C(=O)(CCS(=O)(=O)CC(C)C)N1CC(N(C(C=C)CO)C(C)=O)C1 52621,C1(C(C)NC(c2ccc(C)o2)=O)CCCN(C(c2ccc(NC(C)C)nc2)=O)C1 52622,C1(OC)CCCC(C(=O)NC2(C)CC(NC(c3cc(Br)n(C)n3)=O)C2)C1 52623,c1(C(=O)NCC2(O)CCCN(C(C(C)=C(CC)C)=O)C2)cc2c(=O)[nH]ccn2n1 52624,C(=O)(C(F)C(C)(C)O)NC(C(C)C)CNC(=O)C=Cc1ccccn1 52625,c1(CNC(C(C)c2ccsn2)=O)ncoc1CCNC(C1CC1F)=O 52626,Cc1cc(F)ccc1C(O)C(=O)NC(C)CC(c1ccc(F)cc1)O 52627,N1(C(c2n[nH]c(C)c2O)=O)CCC(CNC(=O)Cn2cc(Br)cn2)C1(C)C 52628,C(=O)(C=CSc1ccccc1)NCCN(C(c1nscc1N)=O)CC 52629,Nc1ccc(C(N2CCCCC(CNC(=O)COCC(F)(F)F)C2)=O)nc1F 52630,N1(C(C2C(CC)CCN2C(C2CC3CCCC23)=O)=O)CCSC2(CCC2)C1 52631,N1(C(COCCCC)=O)CC2CCN(C(C3CCCCS3)=O)CC12 52632,N1(C(C(F)OC)=O)CC(C2CCCCN(C(c3ncc(C)cc3F)=O)C2)C1 52633,C1(CC(=O)N(CC(C)(C)CNC(c2ccc(Cl)s2)=O)CC)C(=O)N(C)N=C1C 52634,N1(C(CS(=O)(=O)NC)=O)CCCC(C)(C)C1C(=O)NC1CN(C)C(C)(C)C1 52635,C1(NC(c2cn(CC(C)C)nc2)=O)COCCN(C(c2ccc(=O)n(C)n2)=O)C1 52636,c1(C(=O)NC2CCC(CNC(c3nocc3Cl)=O)C2)ccc(F)c2cnccc12 52637,c1(CC(=O)NCCCNC(C2C3CCC(=O)C23)=O)ccc(F)cc1Br 52638,N1(C(CNC(=O)OCC=C)=O)CCCC1C(C)NC(C1(C(F)F)CC1)=O 52639,C1(NC(c2cnc(C)[nH]2)=O)C2CCC(C2)C1C(N1CCC(O)C(F)C1)=O 52640,C(CNC(=O)C(C)CC1CC1)(C(C)(C)C)NC(c1c(OCC)scc1)=O 52641,c1(N2C(C)C(N(C)C)CC2)cc2ncn(Cl)c2cc1C#N 52642,C(=O)(C(C)Cn1ccnc1)N(C)CC1(NC(CCN(C(C)=O)C)=O)CC1 52643,C(c1ccc(F)c(F)c1)=C(C(=O)N(CCNC(CCOC(C)=O)=O)C(C)C)C 52644,c1(C(N(C(C(=O)OC)C)CC)=O)cc(C2CC2)ccn1.c1(C=O)cccc(O)c1 52645,Cn1nc(Cl)c(C(=O)NCC2CCCC2NC(c2cncc(F)c2)=O)c1Cl 52646,C1(C(=O)NCCc2ccncc2)(COC)CN(C(=O)CCC2CC2(C)C)C1 52647,C1(C(N(CCCCN(C(C(CCN(C)C)N(C)C)=O)C)C)=O)CCCC(=O)CC1 52648,C1(CNC(CCC)=O)(CNC(=O)CC(c2ccc(Cl)cc2)O)CC12CCC2 52649,C(=O)(C(C)(C)NC(=O)OC(C)(C)C)N1CC(C(C(=O)NCC2C(C)C2)O)C1 52650,C1(C)(CC(=O)N(CC)CC2CCCN2C(=O)CC#N)CCCCC1 52651,CC(C(=O)N1CCC(C)(C(=O)NCCOC2CCCC2)CC1)S(C)(=O)=O 52652,S(=O)(=O)(c1cc(Cl)ccc1F)N1C(C(=O)Nc2ncc(OC)cc2F)COCC1 52653,CS(=O)(=O)c1ccc(C(=O)NCC(C2CC2)NC(C2(CO)CC2)=O)o1 52654,C#CCC(C)(C(=O)NCc1cnc(O)c(F)c1)NC(c1cnccc1C)=O 52655,C1(NC(c2c(C)cccc2)=O)CN(C(=O)CC2CNC(=O)C2)CC(C)(C)C1 52656,C1(NC(C=CC=CC)=O)CC2CCC1CC2NC(c1ccncc1O)=O 52657,N1(C(C2C(C)C2)=O)CCN(C(C2CC3CC2C3)=O)C(CS(C)(=O)=O)C1 52658,CCS(=O)(=O)c1ccc(CC(=O)NCC2CN(C(=O)C(C)N(C)C)C2)cc1 52659,C=CCCC(F)(F)C(=O)N1CCC(N(C(=O)CCN(C)CCO)C)C1 52660,C(=O)(C(O)CCNCCC1CCC(=O)N1)NC(C1CCCC(=O)N1)=O 52661,c1(C(=O)NCCCNC(C2C(C)(C)OC(=O)N2)=O)cnn2c(Cl)cccc12 52662,N1(C(C2CCC(C)CC2)=O)CC2(CO)CC1(C(=O)NC1CCN(C(C)(C)C)C1)C2 52663,N1(C(c2c(C)nsc2C)=O)CC(CC(N2CC(N(C)C)C(C)C2)=O)C2(CC2)C1 52664,Cc1ccc2c(C(=O)NC(C3CCCN3C(c3c[nH]c(=N)s3)=O)C)c[nH]c2c1 52665,C(C)(C(CC(=O)NCc1noc(C)n1)NC(c1[nH]cc(C)c1C)=O)OC 52666,C(=O)(C(C(C)C)C(C)C)N1C(CNC(C2CCCC(=O)N2)=O)CC(OC)C1 52667,CCCC(CCO)ONC(C1CCCN(c2ccc(NC)cc2)C1)=O 52668,N1(C(c2c(CC)scc2)=O)CCOC(CCNC(=O)CCCn2cccc2)C1 52669,C12(NC(=O)C(c3cccc(Br)c3)O)CCC(C(N3CC4(CCC4)C3)=O)(CC1)CC2 52670,C(C)(C)(CCC(=O)NC1CCN(C(c2cc(F)cs2)=O)CC1C)OC 52671,Cc1cc(NCc2ccc(S(N)(=O)=O)cc2)ncc1S(=O)(=O)NCCS(C)=O 52672,c1(C(N2CCC(O)(C(CNC(C(C)=C3CCC3)=O)C)C2)=O)cnc2scc(C)n12 52673,CS(=O)(=O)C=CC(=O)NCC1(O)CCN(C(C2CC3(CCC3)C2)=O)C1 52674,c1(C(=O)NC2C(C)N(C(c3cn4c(n3)SCC4)=O)CC2)cc(F)c(Cl)cc1Cl 52675,Cc1c(Cl)ccc(CCNOCC(CC(C)CO)O)c1Cl.c1(C)ccco1 52676,c1(C(N2C(C)(C(=O)Nc3cncc(OCC)c3)CC2)=O)ccc(F)c(F)c1 52677,C1(SCC)CC(CC(=O)NC2CC(NC(=O)C(Br)=C(C)C)C2)C1 52678,Cc1ncc(C=CC(=O)NC2CCC(CCNC(=O)CCS(N)(=O)=O)C2)c(O)n1 52679,C(=O)(CN1C(=O)CCOc2ccccc21)NCC1OCCN(C(C)=O)C1 52680,C(c1ccccc1)=C(CC)C(=O)NC1(CNC(c2cc(Cl)ccn2)=O)CCC1 52681,c1(C(=O)NC2C(NC(Cc3c(C)scc3)=O)CCOC2)ccc(N)c(Cl)n1 52682,c1(OC)cccc(N(CCCC2CCCO2)C)c1NC(c1ccccc1)=O 52683,Cc1ncc([N+](=O)[O-])cc1C(=O)NCCCCN(C)C(C1(C(C)(C)O)CC1)=O 52684,C1(C(=O)O)CC(F)(CNC(C2C=CCCN2)=O)C1 52685,CC1C(=O)N(CC(N2CC(NC(=O)C=CBr)C3(CCC3)C2)=O)C(=O)C1C 52686,N1(C(CN2CC(C)(C)C2)=O)CCCC(C(=O)NCc2cncc(Cl)c2)CC1 52687,C1(NC(c2cc(C)[nH]n2)=O)COC2(CCN(C(C3(CO)CCOCC3)=O)C2)C1 52688,CCCS(=O)(=O)CC(=O)NCC1CC2(CO1)CN(C(c1c(C)ncn1O)=O)C2 52689,c1(-c2n(-c3cccc(C)c3)nc(C3CCOC3)n2)cn(C)cc(Br)c1=O 52690,c1(C(=O)OCC)ccc(CSc2cc(-c3ccccc3)n[nH]2)cc1 52691,CCC(C)(C)CC(=O)NCCCC1CCCN1c1nc(Cl)ncc1Br 52692,N1(C(C(C)NC(N)=O)=O)CC(O)(C2(CNC(=O)CC(C)(C)O)CC2)C1 52693,c1(NC(C)C)ccc(C(=O)NCC2(O)CN(C(C3CC3(C)Br)=O)C2)cn1 52694,c1(C(=O)NC(CC(=O)N(C)CC)C)ccc(OC)c(C#N)c1F 52695,c1(NC(CNC(c2ccn(C(CC)CC)n2)=O)C2CC2)cc(O)nc(O)n1 52696,C1(NC(c2cc(CC)sn2)=O)CC12CCN(C(=O)C(C)C1CCCC1)C2 52697,N1(C(C(C2(O)CN(C(c3ccc(OC)o3)=O)C2)F)=O)CC(=O)NCC1C 52698,N1(C(c2cc(C)oc2)=O)CC(NC(=O)C(C)Cc2cnc[nH]2)C(N=[N+]=[N-])C1 52699,C(C(F)(C(=O)NC(CC)C(N)=O)C(C)C)NC(c1ccn(CCC)n1)=O 52700,c1(NCC(CNC(C2CC=CC2)=O)O)cc2nncn2cn1 52701,n1(CC(C)NC(=O)CCc2ncc[nH]2)cc(CNC(=O)C(C)(F)F)nn1 52702,c1(-c2n(-c3c(CC)cccc3)nc(C(O)CC)n2)ccc(F)c(Cl)c1F 52703,c1(C(N(C)CC2CCN(C(=O)C=CC3CCOCC3)C2)=O)cn2c(n1)CCCC2 52704,N1(C(C=NOC)=O)Cc2nccn2CC(NC(c2cccc(C(F)(F)F)n2)=O)C1 52705,c1(C(N2CCCC(n3cc(C(C(C)C)O)nn3)C2)=O)ccc2ncn(C)c2c1 52706,C1(C)(CCNC(C(N2CCCCC2=O)C)=O)CCN(C(=O)Cn2ncnn2)C1 52707,Cc1cc(C(=O)NCCN(CC(C)O)C(=O)CSS(C)(=O)=O)c(O)c(C)c1 52708,N1(CCNC(C2(CCNC(c3cccc(CO)n3)=O)CC2)=O)CCNC(=O)C1 52709,c1(OC)cc(Br)c(CNC(=O)C(C2CCS(=O)(=O)CC2)F)cc1C 52710,c1(OC)ccc2cc(C(N3CCC4(CCN(C(=O)C5CC5)CC4)C3)=O)n(C)c2c1 52711,N1(C(c2c(C)nc(CO)nc2)=O)CCN(C(c2ccccc2O)=O)CC12CCC2 52712,C1(CCC(=O)NCC2(Cl)CCC2)CCCCN(C(c2ccc[n+]([O-])c2)=O)C1 52713,C(=O)(CCCCC(F)F)NC(C)CCNC(C1(CF)CCOCC1)=O 52714,N1(C(c2ccccn2)C)CCCC(C)(CN=c2[nH]nc(C(F)(F)F)s2)C1 52715,CC1CC(NC(c2ccnn2C2CCOCC2)=O)CN1C(=O)C=C1CC1 52716,N1(CCCNC(CC=CC)=O)CCN(C(c2cccc(C3CCC3)c2)=O)CC1 52717,C(F)(F)(C(F)(F)F)Oc1ccc(N2CCC(C(=O)OCC(F)(F)F)C2)cc1 52718,c1(C(=O)NC(CN(C(C2(COCC)CC2)=O)C)(C)C)ccc(N)c(C)c1F 52719,n1(CC)nc(C(=O)NC(C2CN(C(=O)Cc3ccncc3Cl)CCO2)C)cc1C 52720,Cc1[nH]nc(CO)c1C(=O)NC1CC(C)N(C(=O)CCN(C2CCCCC2)C)C1 52721,C1(C(=O)NC2C(NC(CN(C)C(c3cccs3)=O)=O)CCC2)Cc2cscc2C1 52722,C1(NC(c2ccc(F)c(Cl)c2F)=O)CCC12CCN(C(C1CCC(O)C1)=O)CC2 52723,c1(C(N2CCC(Oc3ccccc3F)CC2)=O)ccc([N+](=O)[O-])[nH]1 52724,CC(Cn1cccn1)C(=O)N(C(C)C(=O)NCCc1ccn(C)n1)C 52725,C1(NC(CC2CC(N(C)C)C2)=O)CCN(C(=O)CCc2n[nH]c(=N)s2)C1 52726,N=c1cc(C(N2CCN(C(C3CC=CCN3)=O)CC2)=O)cc[nH]1 52727,C1(C)(C(=O)NC(C)C(C)NC(C2(CO)CCCC2)=O)SCCCS1 52728,C#CC1C(C(N2CCC2CNC(=O)CN2CCC(O)CC2)=O)C1(C)C 52729,C(=O)(CC(O)CC(C)C)N(CCOC)CCNC(=O)Cn1nc(C)nc1C 52730,Cc1c(C(=O)NC23CCC2CN(C(c2cc(Br)n(C)n2)=O)C3)nn(C)c1N 52731,Cc1c(Br)csc1C(N1CCCC1Cn1cc(C2OCCO2)nn1)=O 52732,n1(CC(=O)NCC2C(NC(C=C(C)C3CC3)=O)COC2)ncn2nccc2c1=O 52733,c1(CC(N2CCC(CCNC(CN3C(C)CCC3)=O)C2)=O)ccccc1C(C)C 52734,N(C(=NCCC1CCC2(CCC2)O1)NCC(c1ccccn1)(C)C)C1C(C)C1 52735,C1(NC(=O)Cc2cncnc2)CC12CCC(NC(c1cc(Cl)cs1)=O)CC2 52736,c1(OC)ccn2ncc(-c3ccnc(NC(=O)C(F)(F)C(O)C4CC4)c3)c2c1 52737,CC1(NC(=O)C(=O)NC(C)(CC(F)(F)F)CO)CCOC1 52738,N1(C(c2sccc2I)=O)CC2CC2(C(=O)NC(CO)C2CC2)C1 52739,c1(C(C(=O)NCCCCCNC(=O)CC(C)c2ccon2)OC)ccc(Cl)cc1 52740,c1(CN2CCC(CCC)C2)cc(NC(c2cn(CC)nc2C)=O)ccn1 52741,C12(C(=O)NCCn3ncc(C(=O)NC(COCC)C)c3)C=CC(CC1)C2 52742,Cc1ccc(C(N2C3CN(C(c4cnn(C)c4C(F)(F)F)=O)CC23)=O)c(F)c1 52743,CCCC(C(=O)N1CC(NC(=O)C=CC2CCC2)CC(F)C1)S(N)(=O)=O 52744,C1(NC(=O)Cn2cc(Br)cn2)CN(C(C2CC3(C2)CC3F)=O)CC12CCC2 52745,C(=O)(CC(C)(C(F)F)N(C)C)NCCN(C(C1(C)CCC(=O)N1)=O)CC 52746,CC12CCC(C(=O)NC3CC(O)CN(C(=O)Cc4ccsc4)C3)(CC1)CO2 52747,CC1CC(C)C(CNC(C23CC(CF)(CO2)C3)=O)CN1C(=O)C1=CCCCC1 52748,c1(CNCCCc2ccc(F)cc2)ccc(F)c(F)c1Br 52749,c1(C(=O)NCCc2n[nH]cc2Br)cn(C(F)F)nc1C1CC1 52750,C(CC(=O)N(C)CC1(CO)CC1)(C(C)(C)C)NC(c1cc(C)c(=N)[nH]c1)=O 52751,c1(C(=O)NCC(C)N(C(C(CC)CCOC)=O)C)cc2c(OC)ccc(C)c2[nH]1 52752,C(=O)(CC(C)N(C(=O)CN(C)C(=O)OCC)C)N(C(CCC)C)C 52753,CN1CCC2C(CCCN2C(COC(C)(C)C)C(=O)NC2(C)CC2)C1 52754,C1(NC(=O)C=Cc2ccncc2)CCCN(C(C2(c3cccnc3)CC2)=O)CC1 52755,O=[N+]([O-])c1ccsc1COC(c1cc(Br)ccc1F)=O 52756,c1(-c2nc(C(C)OC)nn2-c2cc(Cl)nc(Cl)c2)ccc(C)c(NC2CC2)c1 52757,c1(C(=O)NC(C2(CC=C)CCC2)c2cnn[nH]2)cnc(C(F)(F)F)c(C)c1 52758,c1(SC)cn(C)nc1C(=O)NC1CC1CNC(c1ccc(CN(C)C)cc1)=O 52759,c1(C(N2CCCC(C(C)NC(CCOCCC)=O)C2)=O)nnc(O)cc1O 52760,c1(C(=O)NCC(C)NC(COC)=O)ccccc1C(=O)N(C1CCC1)C 52761,C1(COC)CCCCCC1(F)F.c12nocc1C(c1nnnn1C(C)C)N2 52762,N1(C(C=Cc2ncn(C)c2)=O)CC(C2CC2C(=O)NCC2(C3CC3)CC2)C1 52763,c1(CC(=O)N(CC(CNC(C(CCC)OC)=O)C)C)ccc2ocnc2c1 52764,c1(C(=O)NCC2(NC(CCNC(C)=O)=O)CCCCC2)cc2c([nH]1)CCOC2 52765,C(=O)(C1=CCCCC1C)NCC1CN(C(C2(C(=O)OCC)CC=CC2)=O)CC1O 52766,n1(CC(C)C)c(N(C)CC2CCCCC2)nnc1-c1nc(C2(C)CC2)no1 52767,C1(NC(C=COCC)=O)(CNC(C2CCCS2)=O)CCC(C)(C)CC1 52768,CC1(C)CCN(C(C2(C#N)CC2)=O)CC1NC(=O)CCCOCc1ccccc1 52769,O=C1CC(C(=O)NC(c2cccc(F)c2)c2ccccc2)=NN1 52770,N1(C(c2ccc(C#C)nc2)=O)CCN(C(C2CC2(F)F)=O)CC(O)C1 52771,C1(NC(Cc2nc(C)[nH]n2)=O)CC(=O)N(C2CN(CCC(=O)NC3CC3)C2)C1 52772,CC(C)C(C(=O)N1CCCC1CCNC(=O)C(F)OC(F)(F)F)NC(N)=O 52773,Cc1ccc(C(CNC(c2cnc(S)n2C2CC2)=O)NC(=O)CC(C)F)cc1 52774,C1(C(N(C(CC(=O)OC)C)C)=O)(NC(=O)CCn2ccnc2C)CC(F)(F)C1 52775,C12(CNC(C(CCC)OC)=O)CC(CO1)N(C(=O)CCC1CCCOC1)C2 52776,CCCCCCCCC(CCCCCC)C(=O)NCC1CCN(C(=O)CC)C1 52777,c1(CCC(=O)NCCCN(C)C(c2ncccc2Cl)=O)ccc2cccnc2c1 52778,C(=O)C1CC1.N(C1=CCCC1)(C=O)CC12CC(C)(C1)C2 52779,N1(C(c2csc(C)c2C)=O)CCC2CN(Cc3ccc(O)cc3Br)CC12 52780,c1(OCC(=O)NCc2cnc(-n3ncc(C)c3)nc2)ccc(S(N)(=O)=O)cc1 52781,Cc1ccc(Sc2nc(-c3cccc(N(C)C)n3)nn2C2CCOC2C)cc1C 52782,N1(C(C2(OC)CC2)=O)CC(CNC(C2(C)CC(F)(F)C2)=O)OC(C)(C)C1 52783,c1(C(=O)NCCN(C(CS(CC)=O)=O)Cc2ccccc2)cc(C#N)cc(C)n1 52784,C(c1ccc(Br)s1)=C(C(c1nnnn1C1CCOC1)NCC(CC)(C)C)C 52785,C1(CNC(=O)NC2N(C(CCC)=O)CCCC2)(CO)CC2CCC1C2 52786,CN1CCn2nc(C(=O)NCC3CCN3C(c3cccc([N+](=O)[O-])c3)=O)cc2C1 52787,Cn1cc(CC(N2CCCC2CCC(=O)NC2C=CCC2)=O)nn1 52788,CCC(C)(C(=O)NC1CCC(N(C)C(c2ccnc(C)n2)=O)CC1)C(N)=O 52789,c1(C(N(CC(=O)NCc2c(CC)nns2)CC)=O)ccc(C)n1C 52790,N1(C(C2C(CC)CCC2)=O)CCN(C(c2ccc(C)c(O)c2)=O)CC1C 52791,N(C1CCC=Cc2ccccc21)c1cc(NC(c2ccc(Br)cn2)C)ncn1 52792,C1(N(C)C)CCCN(C(C2CN(C(=O)CC3CCCC4CC34)CCO2)=O)C1 52793,CC1(C)CC(CC(N2CCCC2CNC(C2(c3ccsc3)CC2)=O)=O)C1 52794,Cc1c(CC(=O)NC2CN(C(C3(F)C(C)(C)C3(C)C)=O)C2)oc2ccc(Cl)cc12 52795,C(C)(C(CCc1ccccc1)NC(=O)CCF)NC(c1ccc(C)s1)=O 52796,c1(C(N2CCC(C(NOCC)=O)C2C2CC2)=O)cnn2cccc2c1 52797,Cc1c(C(=O)NCC(F)CNC(=O)C(C)(Cl)Cl)oc2cc(Cl)ccc12 52798,C(=O)(C1=CCCCC1C)NCC(C(=O)NC1CC(CSC)C1)C 52799,N1(C(c2c(CC)nccn2)=O)CC2CCCC2(C(=O)NC2(COC)CC2)C1 52800,C1(NC(Cc2nc(C)oc2)=O)C2CC3C1C3C2C(=O)NC(CF)C(F)(F)F 52801,c1(OC)ccc(C(=O)NCCCCCN(C(=O)C2=CCC(C)CC2)C)c(O)c1F 52802,C1(COC)(NC(=O)CC2(OC)CCC2)CCCN(C(=O)C(C)(C)CCOC)C1 52803,N1(C(CSCC(C)C)=O)CCOC2(CCN(C(=O)CC3CN4CCN3CC4)C2)C1 52804,c1(C(=O)NC(CCN(C(Cc2cc(CC)no2)=O)C)C)c(C)noc1C 52805,S(=O)(=O)(c1ccc(NCCC2(C)OCCO2)cc1Cl)NCCCC 52806,c1(OC(C)C(=O)NC2CCCN(C(=O)CCCF)C2)ccccc1Br 52807,C1(NC(C=C(C)C)=O)CC2(CCN(C(C3CC3c3cccc(F)c3)=O)CC2)C1 52808,N1(c2nc(C)c(Br)cn2)CC(C)CN(C(C2C3CCCC23)=O)CC1C 52809,N1(C(C2C(C)(C(=O)O)C2)=O)CCOCC1Cc1cn(C2CCCC2)nn1 52810,N1(C(C2CCN(C(C=CCC)=O)C(C)C2)=O)CCCN(C=O)CC1 52811,c1(C(=O)NC(CC=C)CNC(=O)C(C)OCCN(C)C)ccc(O)nc1Cl 52812,N1(C(CCCn2cc(-c3cn(CC)nc3)nn2)=O)CCCC(CC(N)=O)CC1 52813,N1(C(C(Cc2ccccc2)NC)=O)CC=C(c2ccnn2C)C1 52814,c1(N2C3CN(C(C(CC)(C)CC)=O)C(CC3)C2)ccc([N+](=O)[O-])c(O)n1 52815,c1(NC)snc(C)c1C(=O)NC1CCC(NC(=O)CCc2ccc(O)nc2)CC1 52816,N1(C(CC=CCC)=O)CC(OC)CC1(C)CNC(c1ccc(C)cc1N)=O 52817,N1(C(c2c(OCCC)cccc2)=O)CCC(NC(c2ccoc2C)=O)C(C)C1 52818,N1(C(c2c(Cl)ccc(C)c2)=O)CCC2CN(C(C3(C(C)C)COC3)=O)CCC2C1 52819,c1(CN2CCCC(NC(=O)COC(F)(F)C(F)(F)F)CC2)cc2ccccc2o1 52820,Cc1cc(C)c(C(N2CC(NC(c3ccc(F)cc3)=O)C(O)C2)=O)c(Cl)n1 52821,C(=O)(C1=CC2(CCOC2)C1)NCC(CN(C(c1cc(N)c(C)c(N)c1)=O)C)C 52822,CC(C)C(F)(F)CC(=O)N1CC(CNC(c2c[nH]c(C(N)=O)c2)=O)CC1C 52823,c1(SCC(=O)NC2(C)CN(C(c3c[nH]ccc3=N)=O)C2)ccsc1[N+](=O)[O-] 52824,N1(CCCNC(CCN(CC#C)C(C2CC2C)=O)=O)CCCC1C 52825,CC(C)CCCCC(=O)N1CCN(C(c2cccc(-c3nc(O)n[nH]3)c2)=O)CC1 52826,CCCCC(O)CCC(=O)NC(C1CCN(C(=O)CN2CCC(C)CC2)CC1)C 52827,CCCC(O)CC(=O)NCCN(C(=O)Cc1ccc(CC(C)C)cc1)C 52828,N1(C(=O)NC)CCC(NCCCOC(C2CCC2)C)CC1 52829,CC1(NC(c2ncc(Cl)nc2Cl)=O)CCCN(C(c2cscn2)=O)C1 52830,N1(C(c2c(C)cn(C)c2)=O)CCC(O)C(NC(=O)CCN2CCC(F)C2)C1 52831,C1(C(=O)NC2C(C)CN(C(C3(O)CCOC3)=O)C2)CCC2(CCC2)CO1 52832,C(=O)(C(CCOCC)c1c[nH]nc1C(F)(F)F)N(C1CCCCC1)CCC#C 52833,N1(C(C(C)SC(F)(F)F)=O)CCOCC(NC(C2(c3ccno3)CCC2)=O)C1 52834,c1(C(=O)NCc2ccc(C(C)NC(=O)C(O)C(C)C)cc2)cnc(O)n(C)c1=O 52835,N1(C(C(C)CC2CCCC2)=O)CCC(C2CC2)(CNC(=O)COCCF)C1 52836,Cc1c(C(=O)NC2(CCNC(=O)C=Cc3ccoc3)CC2)cc(F)cc1Br 52837,c1(NC(CNC(Cc2cc(C)on2)=O)C(C)C)ncnc2sccc12 52838,C1(C(=O)NCCN(C(C2CC2F)=O)CC)(CO)CCCC1 52839,Cc1nnc2cc(NCCN(C(=O)Cc3cccc(Cl)c3F)C)ncn12 52840,C1(NC(CN(C(C(C)C)=O)C)=O)CCC12CCCN(C(=O)C(F)C(C)(F)F)C2 52841,C1(NC(CS(C)(=O)=O)=O)CN(C(=O)C(=Cc2cccc(F)c2)F)CCC1O 52842,C1(NC(c2nc(CCC)oc2)=O)C2CC3CN(C(=O)CC4=NNC(=O)C4)C1C3C2 52843,CC(CC(=O)N(CCNC(=O)CCC1CC(F)(F)C1)C1CC1)c1c[nH]cn1 52844,c1(CC(=O)NCC(CO)NC(=O)CCc2nncs2)c[nH]c2cnc(Cl)cc12 52845,Cc1ccc([N+](=O)[O-])c(NCC2CC(CNC(C3(C(F)F)CCCO3)=O)CO2)c1 52846,C(=O)(C1=CCCCC1P(C)(C)=O)N1CC2(OCCN(C(C(C=C=C)C)=O)C2)C1 52847,c1(C(=O)NC(c2cn(Cc3ccc(Cl)nc3)nn2)C)cn2ccccc2n1 52848,c1(NCc2cn(-c3ccc(C(C)(C)C)c(Br)c3)nn2)ccc(C#N)c(F)c1 52849,C1(C(=O)NCCCNC(=O)CC2CCCO2)(Cc2cccs2)CCCCC1 52850,C(CNC(=O)CNC(=O)C(N1CCCC(C)C1)=O)(C(F)(F)F)OCC 52851,c1(C(N2CC(C(C(=O)NC(C(C)C)C3CC3)OC)C2)=O)cc(O)cc(=O)o1 52852,C1(C(N2C3CCC2CN(C(C2(C4CC4)CCC2)=O)C3)=O)COC2CCCCC12 52853,N1(C(c2c(C)nc(CSC)s2)=O)CCC(NC(=O)C(C(C)C)NC(C)=O)C(O)C1 52854,CC1(C)CCC(C(=O)NC(C2CCN(C(c3cccc(N)c3)=O)CC2)CO)C1 52855,C1(C(=O)NCC2(C)N(C(c3c(C)nn[nH]3)=O)CCC2)CC12CCCCCC2 52856,Cc1ccc(F)cc1C(N1CCN(C)CC1CNC(c1nccn1C(C)C)=O)=O 52857,n1(CCC)ccc(C(=O)NCCCCN(CCCNC(C2C=CCS2)=O)C)n1 52858,C12(CNC(CCCN(C)C)=O)CCC(CC1)CN2C(=O)C(c1ccc(F)cc1)O 52859,c1(SCCC(=O)NC23OCCC(C(=O)OC)(C2)C3)nc2ccccc2s1 52860,N1(C(c2c(Cl)ccc(C)c2)C(=O)NC2CCC2)CCCC1C1CCCO1 52861,C(C(F)C(=O)NOCCC(F)F)C1CN(C(CCc2n(C)ccc2)=O)C1 52862,C1(C(N2C(C)(CCC(=O)NCCN3C(C)CCCC3)CCC2)=O)CC2CCC(C1)C2 52863,Cc1ccc2[nH]c(C(=O)NCC(O)CCNC(=O)CCC(C)C)cc2c1 52864,C1(NC(C(C)SC)=O)CCN(CC2CCCCO2)C(C)C1 52865,N1(C(c2c(C)n(C)cn2)=O)CCCC(C)(C)C1C(=O)NC(c1nncn1C)C 52866,C1(NC(CCC2C(C)=NNC2=O)=O)CCSC12CN(C(c1ccn(C)c1C)=O)C2 52867,c1(C(N2CCCC(C)(NC(C3C(C)C3)=O)C2)=O)cncc2ccsc12 52868,c1(OC)ccc(-c2n[nH]cc2CN2CC(C(=O)OC)CC(CN(C)C)C2)cc1Cl 52869,N1(C(c2ccc(O)c(O)c2)=O)CC(C(N2CC3COCC3C2)=O)CC(F)(F)C1 52870,c1(NC(c2[nH]cc(COC)c2)=O)cccc(NC(C2(C)CCCO2)=O)c1 52871,N1(C2c3ccc(cc3)NC2=O)CCOC(C(F)(F)F)C1(C)C.CCCCCCOC 52872,c1(Nc2cc3c(cc2)OC(C)C3)nccc(=NC2CCCn3nccc32)[nH]1 52873,N1(C(c2csnc2Cl)=O)CC2OCCN(C(C3CCCN4CCCCC34)=O)C2C1 52874,C1(NC(C2(CNC(C(C)=C3CC3)=O)CCCCC2)=O)CC(O)C12CCC2 52875,C1(C(=O)NCC2(NC(CCNS(CC)(=O)=O)=O)CC2)CC12CCC1(CC1)CC2 52876,c1(CCOC)cccc(CNC(=O)C(c2ccc(Cl)cc2)N(CC(=O)OC)C)c1 52877,C1(NC(CC2CCC(C)CC2)=O)CC2CN(C(=O)CC(=O)NCC3CC3)CC12 52878,c1(OCC)ccc(NC(=O)CN2CCC(c3ccccc3F)C2)cc1 52879,C1(NC(c2cc(C)no2)=O)CCCCC1C(=O)N(C)CC1(N(C)C)CC1 52880,N1(C(c2ccc(F)c(C(F)(F)F)n2)=O)CC(CO)c2ccccc21 52881,c1(C(=O)NC(CC)CNC(c2cc(C)c(Cl)cc2C)=O)cc2[nH]nc(C)c2cn1 52882,C1(C(=O)NC2(C#C)CC(F)(F)C2)C(C2CC2)CCN1C(=O)C=Cc1ccoc1 52883,N1(C(c2n(CC)cnn2)=O)CCC2(CCCC2NC(c2ccc(SC)s2)=O)C1 52884,C(C(CC(C)C)NC(c1cccnc1-c1cnn(C)c1)=O)NC(C=CSC)=O 52885,c1(CCC(=O)NCCCN(C(=O)C(F)(F)C2CC2)C)nnc(-c2ccccn2)o1 52886,C1(OC)CN(C(=O)CCC2CCC(C(N)=O)O2)CC1NC(c1cccc(Cl)c1)=O 52887,C1(C(=O)NCCOCCN(C)C(c2ccccc2Cl)=O)COc2ccccc2O1 52888,N1(C(C(c2n(C)cnc2)O)=O)CC2(CCC(NC(c3ccccc3)=O)CC2)C1 52889,C(=O)(CC(C)CC(F)(F)F)NC1CCC(NC(c2nn(CC)c(C3CC3)c2)=O)C1 52890,c1(NC(C2C3(CN(C(Cc4nnc(C)o4)=O)C3)C2)=O)cc(Br)cnc1I 52891,c1(C(=O)NC2(C)C(C(C)=O)C2)ccc(C(=O)N(C)C)cc1 52892,C(=O)(CC1CCc2ccccc21)N1CC(C2CN(C(C(C)(C)C)=O)C2)C1 52893,C(=O)(CS(=O)(=O)C1CC1)N1CCC(N2CCN(C(CC(C=C)(C)O)=O)CC2)CC1 52894,CCCC(C(=O)NCCCCCNC(=O)C=Cc1cn[nH]c1)S(N)(=O)=O 52895,C(=O)(C(C)(C)CCCC(=O)NCC1(O)CN(C(c2c(C)nn(C)c2Cl)=O)C1)OC 52896,C1(CNCC(c2ccc(Br)cc2)C)CCC2(C1)CC2(F)F 52897,C1(CS(C)(=O)=O)(C(CN2CC(N(C)C)C2)=O)CCCC1 52898,C1(NC(C2CNC(=O)N2)=O)CN(C(C2(C3CC3)CC2)=O)CC12CC2 52899,Cc1nc(C(N2CCN(C(c3c[nH]cc(F)c3=O)=O)CC2C(C)C)=O)cc(O)n1 52900,c1(C(=O)NCC2CCN2C(=O)CC2CC3CCC2CC3)c(F)cc(F)cc1Cl 52901,CC(N=c1ccc(Br)c(S(=O)(=O)N2CC=C(Br)CC2)[nH]1)c1cccc(F)c1F 52902,N1(C(C(CC)(C)O)=O)CCCC2(C1)CN(Cc1cccc(Cl)c1)CCO2 52903,N1(c2c(OC)cncn2)CCC2(CC1)OCCCC2NC(C1CCC(=O)NC1)=O 52904,C1(CNC(CCC)=O)CN(C(C2CCCCC23CC3)=O)CC12CCC2 52905,N(C(=NCCCF)NCCCS(=O)(=O)Cc1ccccc1)C1CC(OC)C1(C)C 52906,C#Cc1cccc(OC2CCN(C(C3CCN(C(=O)C(C)CC)CC3)=O)C2)c1C 52907,c1(C(=O)OC)cc2n(n1)CCCC2NC(C1CCN(C2CCCCC2)C1)=O 52908,C(=O)(C1=CC(C)(C)C1)NC1C=CCN(C(C(c2ccc(N)cn2)C)=O)C1 52909,C(CS(=O)(=O)CC(=O)NCC1CC2CCC1N2C(=O)C(c1ccc(Cl)s1)=O)OC 52910,Cc1cc(C(=O)NC(Cn2ccnn2)C(=O)NCC2(C)CCCC2O)nn1C 52911,C(CC(F)(F)F)(c1ccc(COC)cc1)Sc1cnn(-c2n(CC)nnn2)c1Br 52912,C1(CC)COCC1NC(=O)C(C)(C)NC(=O)C(C)=CC(C)(C)C 52913,c1(C(=O)NCC2N(C(C(CC)OC)=O)CC2)ccc([N+](=O)[O-])cc1C(F)(F)F 52914,N1(C(C(C)Cc2cnc[nH]2)=O)CCC(C)(CNC(=O)CCc2nncs2)C1 52915,C1(NC(c2c(CC)cco2)=O)CC1C1CCN(C(=O)COCCCN(C)C)CC1 52916,c1(OCC)nc(C(=O)NC(C)(C)C(C)NC(=O)C(C)NC(=O)C(C)(C)C)ns1 52917,C(=O)(CC(C)C(C)C(C)C)N1CC(C(C)(C)O)(CNC(C(CCCC)C)=O)C1 52918,C1(C(=O)NCC(CNC(=O)OC(C)(C)C)CO)CC2(C1)CC(N=[N+]=[N-])C2 52919,C12(CNC(c3ccc(-c4ncc[nH]4)nc3)=O)CC1CN(C(c1coc(O)n1)=O)C2 52920,c1(C(C2CCC2)N(c2nc(OC)c(F)cn2)C2CNCC2(F)F)cc(Br)c(F)cc1Cl 52921,C1(C(N2CC3CCCC3C2)=O)CN(Cc2cc(Br)ccc2Br)CCC1(F)F 52922,C1(NC(N(C2CCCC2C#N)CC(C)C)=O)CC2C=CC1CC2 52923,c1(OC)ccc(Br)c(C)c1C(=O)NC1CCN(C(c2cc(C)c(C)cn2)=O)C1 52924,N1(C(CCn2ccc(C)n2)=O)CCC2(CC(NC(=O)CCCOC3CC3)C2)C1 52925,C1(C(N2CCCC(N(C)C(c3scnc3Cl)=O)C2)=O)CCc2cncn2C1 52926,c1(COC)cc(CC(=O)NCC(C)N(C)C(c2c[nH]nc2C(C)C)=O)no1 52927,C(=O)(C(C)(C)C(F)F)N1CC(OCCNC(c2cc(C)c(C)s2)=O)C1 52928,c1(NCC(=C)C)cc(N2CCCC(OCC)C2)nc(C(F)(F)F)n1 52929,N1(C(c2n(C)nnc2)=O)CC2(CC2)CC1CC(=O)NCC1(C)CC1(F)F 52930,CC1CN(C(=O)C(C)(C)N2CCOCC2)CC2(CCN(CC(=O)NCC#N)C2)O1 52931,N1(C(C2(CF)CCN(C(C(C)C#N)=O)C2)=O)C2CCC1CC1(C2)N=N1 52932,C(=O)(CCCN(C)C)N(C(C)C(=O)NCC1(CO)CCCC1)C 52933,CC(C)C(O)CC(=O)NC12CC(NC(=O)CCC3(C)CC3(F)F)(C1)C2 52934,c1(CCC)nc(=NC(CNC(=O)C(C2CCCCCC2)OC)CO)s[nH]1 52935,CC1(CNC(=O)CCCCNC(N)=O)CCCN(C(=O)C(F)OC(F)(F)F)C1 52936,c1(C(N2C(C)(CCC(=O)NC(CCC(=O)OC)C)CCC2)=O)cn2ccccc2n1 52937,c1(-c2cncc(NC(c3c(C(C)=O)c(C)ccc3)=O)c2)c(F)cc(CO)cc1F 52938,c1(C(C(=O)NC2(NC(C3C=CCC3)=O)CC2)O)cc(F)c(F)c(F)c1 52939,C1(N(C(c2c(COC)ncs2)=O)C)CC2CCC(C1)N2C(c1ccc(F)s1)=O 52940,C1(CNC(CC2(CSC)CC2)=O)CN(c2ncns2)CCC12CCOC2 52941,C(=O)(N=c1cc[nH]cc1Cl)NC(C1(F)CC1)C 52942,N1(C(CC=CC=C)=O)CCCC2(C1)CN(C(=O)CC1CCCOC1)CCO2 52943,CC(C(=O)NC(CNC(=O)CCCn1c(O)nnc1O)C(C)(C)C)C(C)(F)F 52944,C1(NC(C)=O)CN(C(C2CCC(Nc3cc(OC(C)C)ncn3)O2)=O)CC1F 52945,c1(C(N2CCCC(CN(C(c3c(CC)nc[nH]3)=O)C)C2)=O)ccnc2[nH]nnc12 52946,c1(CC)nn(C)c(NC(=O)NC2CC2c2cccc(F)c2F)c1Cl 52947,Cc1cc(C(=O)NC2CC3CCC2(NC(C2CC(C)(C)C2)=O)C3)nc(O)c1 52948,C1(C(N2CC(C)=C(C)CC2)=O)N(C(c2cn(C3CC3)cn2)=O)CC12CCCC2 52949,O=C1C2CC3C1C3C2C(=O)NC1(C(=O)NCC2CCC(F)(F)C2)CCC1 52950,C1(CNC(Cc2cnn(C)n2)=O)CC2(CO1)CN(C(c1nc(Cl)ccc1N)=O)C2 52951,N1(C(c2c(Cl)ccc(Cl)c2)c2ccccc2)CCc2c(CBr)cccc21 52952,CC1=C(C(=O)N2CCCC(Cc3ccccc3-c3cc(C)cc(C)c3)C2)CCC1 52953,C1(C(=O)NC(COC)C2CCC2)(C(=O)NCC2(SC)CC(=O)C2)CCCC1 52954,C(=O)(CC(C)CN(C)C(=O)NCc1cc(C)nn1C)OC 52955,C1(C(=O)OC(C)Cc2ccc(Cl)cc2)CCC(=O)C(C)C1 52956,C(CCCCCNC(C1OC2CCC1C2)=O)n1cc(-c2cc(C(=O)OC)on2)nn1 52957,c1(CC(=O)N(CCCNC(=O)CCSC(F)(F)F)CCO)ccc(Cl)nc1 52958,N#CC1CCCC1NCCNS(=O)(=O)NC1CC1 52959,CC1CN(C(C23CC2COC3(C)C)=O)CCN1C(c1[nH]cnc1C#N)=O 52960,CCCCC(C)C(=O)N1CC2(CC2)CC1CNC(=O)C(C(C)O)N(C)C 52961,C1(CC)CCCCC1C(=O)NCc1ccc(CNC(C2CCCC(=O)N2)=O)cc1 52962,C1(NC(C(C=C)C)=O)CC2CC1CC2C(=O)NOCc1ccccc1Br 52963,c1(C(=O)NCC2(NC(CCCCSC)=O)CCOC2)ccc(F)c(Cl)c1 52964,C1(CNC(c2c(CC)nccc2)=O)CN(C(C2CCC(C)CO2)=O)CCN1C 52965,Cc1cc(C(=O)N(C2CCN(C(=O)CSc3n[nH]c(=N)s3)CC2C)C)nnc1C 52966,C(=O)(C1CCCc2nncn21)NCCN(C(=O)C(C)n1ccnc1)CC 52967,C1(N(C(C2(CN(C)C)CCCC2)=O)C)CCCN(C(C2CNC(=O)C2)=O)CC1 52968,C1(NC(C2(C(C)C)CCC2)=O)CN(C(c2ccc(N)c(Cl)c2)=O)CCC1CO 52969,C(=O)(C(O)CC(C)C)NC(C(=O)NCc1c(C)cccc1)c1ccco1 52970,C1(CN2CCCC(C(N3CCN(C)CC3)=O)C2)CN2CCC1CC2 52971,C1(C(=O)NC2(CC=C)CCC2)CCC(CNC(=O)C=Cc2nc(C)cs2)CC1 52972,C(=O)(C1CNc2ccccc21)NCC(CNC(C(C)OCC)=O)O 52973,C1(N(C(=O)COC2CCCCC2)C)CCCN(C(=O)CCC2CC2(C)C)C1 52974,N1(C(C2CCN(C(c3ccc(C#C)o3)=O)C2)=O)CC2CC(OC)C(C2)C1 52975,C(=O)(CCCC(F)F)N1C(CNC(=O)CC23CCCC2C3)CC(OC)C1 52976,c1(C(=O)NCC2N(C(c3ccc(C)nc3N)=O)CCC2C)ccc2scnc2c1 52977,C(C)(C(O)C(F)F)NC(C(CNC(c1cc(C(F)F)[nH]n1)=O)OC)=O 52978,C1(C(CNC(C2(CC)CCOC2)=O)C)CCN(C(c2cccn2COC)=O)CC1 52979,c1(CC(=O)NCCOCCNC(c2cc(O)cs2)=O)csc(-c2ccsc2)n1 52980,C1(C(C)C)CCCN(C(=NCC2CCN(C)C(=O)C2)NCC2CCCCO2)C1 52981,c1(CCNC(c2c(CC)noc2)=O)cc(F)ccc1C 52982,c1(C(=O)NCCOC2CCN(C(CCNC(C)=O)=O)C2)c(Cl)ccc2c[nH]nc12 52983,Cc1c(C(=O)N(C)CCOCCNC(=O)CN2CCC(C)CC2)cccc1Cl 52984,N1(C(C(C)CN2CCOCC2)=O)CCC2CN(C(c3cc[nH]c3)=O)CC12 52985,c1(CC(=O)OC)ccc(C(=O)NC(C)(C)C(C)NC(C2CC23CCC3)=O)cc1 52986,CCS(=O)(=O)CC(=O)N(CC(CC(C)O)c1ccccc1)C(C)(C)C 52987,c1(-c2ccc(C(=O)NCCSC)s2)ccccc1-c1cnc(F)cc1 52988,CC1CC(C(=O)NCCCN2CCN(c3ccccc3)CC2)C1(C)C 52989,c1(N(C(=O)COC)CCS)cc(C)ccc1C 52990,C1(C(CC)C(=O)N2CC(N(C)C(C3CCCO3)=O)C2)CCC(C)CC1 52991,C1(C(N2CC(NC(CC=CC=C)=O)CC3(C2)CC3)=O)C2Cc3ccccc3C12 52992,C1(C(=O)NC(C2(O)CCN(C(C3(C)CC(F)C3)=O)C2)C)CCCOCC1 52993,N1(C(CC2CCCN(C(CC(CC)(C)C)=O)C2)=O)CCn2ccnc2C1C 52994,c1(C2(NC(c3n(CCC)nnn3)C3CCC3)CC2)cccc(C)c1C 52995,c1(C(=O)NCC23CC(NC(=O)COc4ccsc4)(C2)C3)ccc(F)cc1F 52996,c1(C(N(C(c2ccccc2)CNC(=O)Cc2cscn2)C)=O)cnc(C2CC2)o1 52997,N1(C(CCCNC(N)=O)=O)CC2CCC(C1)N2C(C1CC1c1ccc(Cl)cc1)=O 52998,C1(c2n(C(C(=O)OC)C)nnn2)(NCCS(=O)(=O)CCO)CC2(C1)OCCO2 52999,Cc1cc(F)c(N)cc1C(=O)NC1CC(F)CN(C(c2nnc(O)nc2O)=O)C1 53000,CC(C)CC(C)C(=O)NCC(C1CC1)NC(=O)Cc1nnc(S)n1C 53001,CCCCC(C)CCC(=O)N(C1CC2CNC1C2)C1CC(O)C1 53002,N1(C(c2c(CC)cc[nH]2)=O)CCC(CO)C(NC(C2(CCF)CCC2)=O)C1 53003,C(CNC(=O)CCOCC(C)C)(CC(C)C)NC(C=CCN(CC)CC)=O 53004,N(C(=NCCCCl)N1CCCC2(CC2)C1)CCNC1C(C)Cc2ccccc21 53005,CCCCC(C(=O)NC)NC(=O)CCC1(NC(=O)CCn2cccn2)CCCC1 53006,CN1CCC(C(=O)NC2CCCN(C(=O)CC(C)(C)c3cccs3)C2)C1=O 53007,S(=O)(=O)(c1cccc(F)c1C)NCC1(O)CN(Cc2c(OC)c(F)ccc2)C1 53008,C(=O)(CC(C)CC(F)(F)F)NC1CN(C(c2c(OCC)nccc2)=O)CC12CC2 53009,c1(CC)ccc(C(N2CCNC(=O)C2)C(=O)NCCC2CC2)nc1 53010,C1(NC(CC(C)N2CCCC2=O)=O)C2CC1CN(C(c1ccc(Cl)c(Cl)c1)=O)C2 53011,c1(CCC(=O)NCC(COC)C(=O)OC)cnc2ccccc2c1 53012,N1(C(CCNC(C2(O)CCSCC2)=O)=O)CCC(O)(CO)CC1 53013,c1(C(=O)NCCC2CCCN(C(c3cc(OC)ncc3)=O)C2)cc(C#N)[nH]c1C 53014,c1(C(CCC(=O)NCCCCC(C)NC(CSC)=O)=O)cc(C)ccc1C 53015,CN1CCN(C(C2C3CCC(=O)C23)=O)C(CNC(c2ncc(Cl)s2)=O)C1 53016,C1(NC(CC(C=C)CC)=O)CC2CCC(C1C)N2C(=O)CC1=CCCCC1 53017,c1(C(C)C)ccc(C(=O)NC2CC(Cn3cc(C4(N(C)C)CCOC4)nn3)C2)o1 53018,c1(OCC)cnc(NC(c2cncc(-c3cccc(C#N)n3)n2)=O)c(F)c1 53019,c1(SC)cc(C(=O)N(CC(O)CN(C)C(c2ccc(C)cc2)=O)C)c(Cl)cc1Cl 53020,CCC(C)CC(C)N(C(=O)C(CCOCCO)NC(=O)C=CC(F)(F)F)C 53021,c1(CC(=O)NCC2C(CNC(CC(C=C)C)=O)C2)cccc(O)c1F 53022,c1(C(=O)NC(CN(C(=O)C(C)(C)N2CCCC2)C)(C)C)cccnc1N1CCCC1 53023,C(CC(C)C(=O)NC(CNC(c1coc(CS(C)(=O)=O)n1)=O)CO)=CC 53024,C1(CN(C)C(C2CC2C(F)(F)F)=O)CCCN1C(c1cnc(C2CCCO2)s1)=O 53025,N1(C(CC(COC)C)=O)CCCC2(C1)CN(C(=O)CC(C)CN(C)C)C2 53026,C1(NC(C2N(NC(C)C)CCC2)=O)CCC(N(C(=O)COC2CC2(F)F)C)CC1 53027,c1(C(=O)NC2(C)CCN(C(C3C(C)C3C)=O)C2)cc(O)nc2ccc(F)cc12 53028,CN1C(=O)C(=O)N(CC(=O)NC2CCN(C(=O)Cc3nncn3C)C23CC3)C1=O 53029,C(=O)(N=c1ccn(C2CCC2)[nH]1)C12CC(NC(C(C3CC3)OC)=O)(C1)C2 53030,C(=O)(C(C)CC1CCC1)NCC(CC)N(C(=O)CSCc1cccs1)C 53031,CCC(C)(C(=O)NC(C1CCCCC1)CNC(C1(OC(C)=O)CC1)=O)OC 53032,n1(C(CC)C)ccc(=NC(=O)C(O)CCCNC(=O)C=Cc2cncs2)[nH]1 53033,n1(CCC(=O)NCCCN(C(C(C)=C(C)C)=O)C2CC2)nc(C)cc1C 53034,O=C(CNC(=O)C(CO)OCC1CC1)N=c1ccn(CCF)[nH]1 53035,C1(C(=O)NC(CN(C(=O)C=NOC)CC)C)CCN(c2cnccn2)CC1 53036,N1(C(C2C(C)C2C)=O)CCC(NC(C2(C3CCCO3)CCC2)=O)C1C 53037,c1(NC(=O)NC2CCCN(C3CCCC3)C2)ccc(F)c(Br)c1F 53038,c1(C(=O)NC(C(C)NC(CCc2c(C)noc2C)=O)C(C)C)cc(Cl)ncc1O 53039,C=CCC(CC=C)C(=O)N1CCCC(C)C1CNC(c1cnc(S)nc1)=O 53040,C(CC1CC1)(C(=O)N(C)CCC1CCCN1C)NC(CC1CC(C)C1)=O 53041,c1(OCC(N2CC(CNC(C(n3c(C)cc(C)n3)C)=O)C2)=O)ccc(Cl)c(F)c1 53042,Cc1c(Cl)ccc(C(=O)NC2CCC(N(C(=O)COCC(C)(C)C)C)C2)c1N 53043,c1(C(=O)NC2(CC=C)CCCN(C(=O)OC(C)(C)C)C2)cc(Br)cc(O)c1C 53044,Cc1nc2ccc(C(=O)NC(CNC(C3CC(=O)N(C)C3)=O)C(C)C)cc2s1 53045,c1(C(=O)NC2C=CC(C(=O)Nc3c(CC#N)cccc3)C2)cc(Br)cnc1Cl 53046,C12(NC(CC3(CSC)CC3)=O)CCCC1N(c1nc(C(C)(C)C)ns1)CC2 53047,c1(C(=O)NCC2(CCNC(CC(CC)CC)=O)CC2)[nH]c2cc(C)ccc2c1C 53048,C(CCS(=O)(=O)NCC(=O)NC1(CNC(=O)C=C(C)C(C)C)CCOC1)OC 53049,C#Cc1ccc(OCC(=O)NCCNC(=O)CC2CC(CC)=NO2)cc1 53050,N1(C(C(c2cn(C)nc2)O)=O)CC2CC(C1)C2NC(=O)COCC1CCOCC1 53051,CC(CCCO)N=c1[nH]c(N2CC(C)OC(C)(C)C2)nc2c1SCC2 53052,c1(C(=O)NCC(C)(C2CC2)NC(c2ccnc(C3CC3)n2)=O)cc(F)cnc1O 53053,C1(NC(C(C2CCCC2)OC)=O)CCN(C(C2CCCC(OC)C2)=O)C1(C)C 53054,CC1(C)CC(NC(=O)CC2COCC(C)(C)O2)CN(C(c2coc(CO)c2)=O)C1 53055,Cc1cc(C(=O)Nc2nc(Cl)cc(Cl)n2)cc2nc[nH]c12 53056,c1(OC)ccccc1C1(C(=O)NC(C)CNC(=O)OC(C)(C)C)CCC1 53057,c1(CC)cc(CC(=O)NC2(CCNC(=O)C(C)(C)C3CCCCC3)CC2)n(C)n1 53058,c1(-n2cc(CC3CCN(C(=O)CSC4CCCC4)C3)nn2)ccc(CO)c(F)c1 53059,n1(CC(=O)NCCC(CC)(CC)NC(C(CC)O)=O)ccc(=O)c2ccccc12 53060,Cc1c(C(=O)NCC(C)CNC(C2(C(C)C)CCCO2)=O)cnc2ncnn12 53061,CC(C)(O)C#CC(=O)NC1CN(C(=O)COCC(C)(C)C)CC1(C)C 53062,N1(C(C=C(C)C(F)F)=O)CCCCC(CNC(=O)Cc2nc(C(C)(C)C)cs2)C1 53063,Nc1cc(F)c(C(N2CC=CC(NC(=O)C3=CCCC3)C2)=O)c(F)c1 53064,CC1(C)CN(C(c2ccn3nncc3c2)=O)C(CNC(C2(C)CC2(F)F)=O)CO1 53065,c1(C(=O)NC(CC)CN(C(=O)CCC(=O)N(C)C)CC)coc2c(F)cccc12 53066,CCCCC(CC(=O)NC(COC)CCO)NC(C1(C2(O)CCC2)CC1)=O 53067,C12(C(=O)NC3CN(C(C4(C)CCOC4)=O)C3)CC3CC1(CO)CC3C2 53068,c1(C(=O)NCC2C3CN(C(CCC(N)=O)=O)C2CCC3)cc2cccc(F)c2o1 53069,c1(C(C)C)n[nH]cc1C(=O)N(CCCCCNC(C1CCOC1C(C)C)=O)C 53070,c1(C(N2C(CNC(CC(=O)N(C)C)=O)CC2)=O)cc(CO)ccc1Cl 53071,N1(C(Cc2ccc(C(C)C)cc2)=O)CCN(C(c2ncccc2F)=O)CC1C#N 53072,c1(CC(=O)NCC(CC)NC(c2cc(O)cc(N)c2C)=O)ccc([N+](=O)[O-])cc1 53073,N1(C(C(C(C)C)NC(C)=O)=O)CCCN(C(c2sc(F)cc2Cl)=O)CC1 53074,c1(CCC)cccc(C(N2CC(NC(=O)C3=NOCC3)C(O)C2)=O)c1 53075,C1(O)(CNC(c2cnc(O)c(Cl)c2)=O)CCCN(C(c2ccnn2C2CC2)=O)C1 53076,Cc1cccc(Br)c1C(=O)Nc1cccc(CNC(c2c(C)nn(C)c2C)=O)c1 53077,c1(C(C(=O)OC(c2cccc([N+](=O)[O-])c2)CC)=O)cc2c(cc1Cl)OCCO2 53078,Nc1ccc(C(=O)NC2CC(F)(CNC(C3CCCN3N=O)=O)C2)nc1N 53079,c1(OC)ccc(NC(=O)NCCCOc2c(C)cccc2Cl)c(F)c1 53080,CC(CCO)C(=O)N1CCC1C(N1CC(c2ccc(Cl)cc2)C1)=O 53081,C=CCC(CNC(c1ccc(C#N)cc1)=O)C(=O)N1CC(C)(COC)C1 53082,N1(C(C(=O)NCC)=O)CCC(NC(c2cn(CC(N)=O)nn2)=O)C(F)C1 53083,C1(CN2CCC(CN3CCCCC3)CC2)C2CCC(F)(F)C12.CC(C)C1C(=O)N1 53084,CCCC(CCC)CC(=O)N1CCC(O)C1C(=O)NCC(O)C1(Cl)CC1 53085,C1(CC)CCCN(C(=O)C(COC)CNC(C2CCC=CCCC2)=O)CC1 53086,c1(NC(CC2N(C(C(CC)CC)=O)CC(O)C2)=O)cc(C#N)cnc1C 53087,c1(C(=O)NC(CNC(c2nnc(C)s2)=O)C(C)C)cccc(S(=O)(=O)CF)c1 53088,C1(c2ccccc2)(NC(CC2CC(C)C2)=O)CC(NC(=O)C(C)CO)C1 53089,C1(CC(=O)OCC)CN(C(c2ccn(C(F)F)n2)C(=O)NCC2CC2)CCO1 53090,C1(NC(C(C=CC)O)=O)C(C)(C)C(NC(=O)Cc2cccs2)C1(C)C 53091,C=C(C)CCCC(=O)N.c1(NC(CC)=O)cc(OC)ccc1-c1nnc(C)o1 53092,c1(C(N(CCC)CCNC(c2ccc(OCF)cc2)=O)=O)cc(N)ccc1O 53093,S(=O)(=O)(CC(=O)NC1CN(C(c2cnc(N3CCCCC3C)s2)=O)CC1C)NC 53094,c1(C(=O)NC(CNC(C2CCCC2)=O)C2CC2)cncc(F)c1Cl 53095,N1(C(C(C=CC)O)=O)CC2(C1)CN(C(c1ccc(Cl)cc1C)=O)CC2CO 53096,N1(C(CCCOC)=O)CC(C)OC2(CCN(C(c3c(N)cc(Cl)cc3F)=O)C2)C1 53097,C1(C)(C(N2CC(CN(C)C(C3OCC3(C)C)=O)OCC2)=O)CCCCNC1=O 53098,c1(-n2cc(C3(C)CN(C(Cc4scc(CC)n4)=O)C3)nn2)ccc(Cl)cc1 53099,c1(C(N(C)CCN(C)C(c2cc(C(N)=O)c[nH]2)=O)=O)cc(C(F)(F)F)n(C)n1 53100,CC1=C(C)CC(C)(NC(=O)C(C)CN(C)C(c2cc3ccncc3[nH]2)=O)CC1 53101,N1(C(CCCC=C)=O)CC2(CCN(C(=O)Cc3csc(CC)n3)CC2)C1CCOC 53102,Cc1c(C(N2CCCCC(N(C(=O)C=CCO)C)C2)=O)oc2ccccc12 53103,C1(C(N(CC)CC2CCCN2C(=O)CP(C)(C)=O)=O)OCC2CCCC12 53104,c1(C(=O)OC)nc(C(=O)NCC2(NC(=O)C(CO)N(C)C)CCC2)co1 53105,C(=O)(C(O)CC(C)C)N1CC(N2CCN(C(c3c(C)nns3)=O)CC2)C1 53106,C=CC(C)(C)C(=O)NCCN(C(C1CC1C1CC1)=O)CC1CC1 53107,c1(C(=O)OC)cc(C(=O)NCC(O)CN(C)C(c2ccn(C)n2)=O)c(C)s1 53108,C=CCC(CC)C(=O)NCC1CN(C(c2nonc2CC)=O)CC1C 53109,c1(C(=O)NC2CN(C(COC(C)(C)C)=O)C3C2C3)cc(S(N)(=O)=O)ccc1Cl 53110,N1(C(c2nc(C(C)NC(=O)C=Cc3cc[nH]c3)oc2)=O)CCCC2C1CCN2C 53111,C1(C(=O)NC(CCCC)CNC(c2cc3cscc3s2)=O)CCCC(F)(F)CC1 53112,C1(C)(CNC(COC(C)=O)=O)CCN(C(=O)Cc2sccc2Cl)C1 53113,C1(C(=O)NCC(COC)C)CCN(C(=O)CC2C(C)(C)C2(C)C)CC1O 53114,C1(CNC(CSCc2nc(C)sc2)=O)CC2CCC1N2C(c1ccc(Cl)[nH]1)=O 53115,c1(SC)nn(C)cc1C(=O)NCC1(O)CN(C(=O)C=C(C2CC2)C2CC2)C1 53116,C=CC(C)(O)CC(=O)NCCOC1CCN(C(=O)CCC2CCC(=O)NC2)CC1 53117,N1(C(C)=O)CC(C)(C)OC2(C1)CN(C(c1nn(-c3ccccc3F)cc1O)=O)C2 53118,C1(NC(C(CC)n2cccn2)=O)CCCCCN(C(=O)C=Cc2cnc[nH]2)C1 53119,Cc1ccc(F)c(C(=O)NCC2CC(C)N(C(=O)CSCc3ccncc3)C2)n1 53120,c1(CC)nc(C(N2CCC(O)(Cn3cc(-c4csnn4)nn3)C2)=O)c(C)o1 53121,c1(C(=O)NC2CCN(C(c3[nH]c(=NCC)sc3)=O)C23CC3)cnc2ncccn12 53122,C(CN=c1nc(-c2ccccc2)nc[nH]1)(C1CC1)NC(=O)Cc1ccc(F)cc1 53123,c1(NCC2(F)CCC(C(=O)OC)C2)nc2c(cc1C#N)CCC2 53124,c1(OC)ncc(C(=O)NC2CC(O)CN(C(=O)OC(C)(C)C)C2)cc1C(=O)O 53125,N1(C(=O)Cc2csc(S)n2)CCCCC2(C1)CN(C(C1CC=CCC1)=O)C2 53126,CCC(CC)C(F)C(=O)N1CCC(CC(N2CCCNC(=O)C2)=O)C1(C)C 53127,c1(OC)cc(C#N)ccc1C(N1CCC(C(C)C)CC1)C(=O)NC1COC1 53128,C1(C(C)(C)NC(C2N(CC)CC2)=O)CCN(C(=O)CC2CCC(=O)C2)CC1 53129,C1(C(=O)NCC(CC)(O)CC)CC(N=[N+]=[N-])CN1C(C1CC2CC(=O)C1O2)=O 53130,C(C(=O)NNC(=O)c1coc(-c2ccc(C)cc2)n1)NCC(F)F 53131,N1(C(c2c(C)cno2)=O)CC(NC(c2c(Cl)cncc2Cl)=O)CC(O)C1 53132,C(COC)(N=c1cc(C)nc(NC(C)C2CC2)[nH]1)c1ccc(CC)o1 53133,N(C1CCc2c(Cl)ccc(F)c21)CCCN1CCN(C(C)(C)C)CC1 53134,C1(NC(C=CSC)=O)CCCC(N(C)C(c2cc(N(C)C)ccn2)=O)C1 53135,C1(CC)C(NC(C2(CO)CCCO2)=O)CCN1C(=O)CCC(=O)OC(C)(C)C 53136,N1(C(C=CC(=O)OCC)=O)CCC2(C1)CN(C(C1(C)CCOC1)=O)CCO2 53137,c1(C(CC)C)nc(C)cc(=NC(CCNC(C2CC3(CCOC3)C2)=O)C(C)C)[nH]1 53138,C1(C(=O)Nc2c(OC)cccc2Cl)CCC(N=c2ccn3ncc(Br)c3[nH]2)CC1 53139,C1(CCC(=O)NCC(CC)N(C)C(C2CC(=O)N(C)C2)=O)CCCCN1C 53140,NS(=O)(=O)c1ccc(CN2CC(C(N3CCCC4(CCO4)C3)=O)CC(F)C2)cc1 53141,C1(C)(C(N2CCOCC(NC(CSCCC)=O)C2)=O)CCCNS1(=O)=O 53142,C(=O)(C1CCCc2scnc21)N1CC(O)CCC(NC(c2n[nH]c(C)c2C)=O)C1 53143,N1(C(C(CSC)OC)=O)CCCC(N(C(=O)Cc2cc(C)cs2)CC2CC2)C1 53144,Cc1oc(Cl)nc1C(=O)NCCCCC1CN(C(=O)C(=O)NCC(F)(F)F)C1 53145,C1(C#N)(C(=O)NCC2CN(C(c3c(C)n(C)nn3)=O)C2)CCOCC1 53146,c1(CC(N2C(C(=O)Nc3cc(Cl)ccc3Br)CC(O)C2)=O)c(F)cc(F)cc1F 53147,C1(CC)CN(C(C2(C(N)=O)CC2)=O)CCC1NC(=O)CCc1ncc[nH]1 53148,CC(C)C(F)(F)CC(=O)NC1CCCC1NC(c1cc(Cl)cn1C)=O 53149,c1(CC(=O)C(=O)OC2CN(C(N(C)C)=O)C2)ccsc1[N+](=O)[O-].C1CO1.SC 53150,c1(OC)c(C(N2CCC(C(N3CC(O)C3)=O)C2)=O)cnn1-c1ccccc1 53151,Cc1nc(CCC(=O)NCCC2CCN(C(c3c[nH]nc3C(F)F)=O)C2)cs1 53152,c1(OC)ccc(CN(C)C(=O)NC2CCCOC2c2cn[nH]c2)c(OC)c1 53153,C1(NC(C(NOC)=O)=O)C2CCC1CN(C(=O)COc1cccc(C)c1)C2 53154,C1(CC(N2C(CCC=C)CCC2)=O)CCCCN1C(c1cnnn1CCOC)=O 53155,CC1CN(C(=O)C(C)(C)C(F)(F)F)CC(C)C1NC(=O)C(c1ccc(F)cc1)=O 53156,N1(C(COCC(=C)C)=O)CCC(C)(CCNC(=O)CCc2cc(Cl)no2)CC1 53157,c1(C(N2C(C)CC(CNC(CC3CC(=C)C3)=O)C2)=O)ccc2nccn2n1 53158,n1(CC)nnc2c(NCC3(NC(=O)CC(C)(O)C4CC4)COC3)ncnc12 53159,C1(CC(=O)N(C2CCN(C(COCCOCC#C)=O)C2)C)CCCN(C(C)C)C1 53160,N1(C(c2ccc(C(C)=O)[nH]2)=O)CCC2CCN(C(c3ncccc3Br)=O)C2C1 53161,C1(O)(C(=O)NCC(N(C(=O)C(C)(C)c2ccccc2)C)C2CC2)CC2CCC1C2 53162,C1(C(=O)NCC(CN(C(C2(CC=C)CC=CC2)=O)C)O)CC(F)(F)C1(C)C 53163,c1(C(=O)OC(C#C)C)ccc(-n2nc(C)cc2C)c(F)c1 53164,c1(C(=O)NCC(Cn2cc(CN3CCC(=O)CC3)nn2)OC)ccc(F)cc1Br 53165,c1(OC)cnc(C(N2CC=CC(C(N3CCC3C(=O)N(C)C)=O)C2)=O)cn1 53166,CC1(C)C(C(N2CC(O)(CNC(=O)C(F)=C3CCCC3)C2)=O)C1(F)F 53167,C1(NC(c2scc(OC)c2)=O)COCCN(C(=O)C(F)(F)c2cnccn2)C1 53168,C(=O)(C(O)C(F)F)OC(CC(C)C)C.C1CCC(C)NC(=O)O1 53169,N1(C(c2ccc(CC)nc2)=O)CCCC(NC(c2cn[nH]c2)=O)C1C 53170,c1(N2CCC(Cn3c(C)nc(C)n3)C2)nc(=N)[nH]c(=NCC2=COCCO2)[nH]1 53171,N1(C(C2=CCCC2C)=O)CCC(C(=O)NCC2CC3CCCC3C2)C12CCC2 53172,c1(C(=O)NC(C)C(C)NC(C2(CCO)CC2)=O)cnc(-c2ccccn2)nc1 53173,N1(C(c2n(C)ccn2)=O)CCCC1(C)C(=O)NCC1(c2ccccc2)CCCO1 53174,C#Cc1ccc(C(=O)N(CCC(=O)NCC2CC2C(N)=O)C)c(C)c1 53175,N1(C(C23C(C(=O)OC)(CCC2)C3)=O)CCCCC(NC(C2(C)CC(C)(C)C2)=O)C1 53176,c1(OC)c(C(=O)NCCC(C)NC(C2(C)COC(=O)C2)=O)cnn1C 53177,C1(NC(C2N(C(C3N(C)CC(O)C3)=O)CCC2)=O)CCCCC1(C)O 53178,N1(C(=O)C=Cc2ncc[nH]2)CCCC2(CNC(C34CCN(CC3)C4)=O)CCCC12 53179,C(CCC(=O)NCC1CCCCC1)(C(C)C)NC(c1nccc(C)c1N)=O 53180,Cc1ccc2c(N(C3CC(N)C3)C(c3ccc(Cl)cc3CO)=O)ncnc2c1 53181,c1(C(=O)NC(C(C)C)CCNC(=O)C(C)C2CC2)cccc2nc(C(F)F)[nH]c12 53182,n1(CC)cc(C(=O)NCC(C)NC(=O)CCC2NC(=O)NC2=O)c2ccccc12 53183,c1(C(=O)Nc2c(C(=O)OC)cc(Br)cn2)cn2c(n1)CN(Cc1cc[nH]c1)CC2 53184,N1(C(CSCC)=O)CCc2ccccc2C(NC(=O)CC2(COC)CC2)C1 53185,c1(CNC(=O)CC2(O)CNC2)ccc(CNC(=O)C(c2ccccc2)F)cc1F 53186,CCC(C)(C)C(C(=O)NCC1(CNC(=O)C(C)(COC)OC)CCOCC1)OC 53187,c1(C(C)NC(c2c(C#C)c[nH]n2)=O)cc2ccccc2n1C 53188,C1(CC(=O)NC2C=CCN(C(c3ccc(CC)o3)=O)C2)NC(=O)CN(C)C1=O 53189,C1(F)(CNC(C2Cc3nncn3C2)=O)CCCN(C(C2(CO)COC2)=O)CC1 53190,c1(N2CCC(CCC)C2)nc2ccccc2c(=NCC(F)(F)Br)[nH]1 53191,C1(C(=O)NCCOC2CCN(C(c3cc(F)cs3)=O)C2)CCc2nc[nH]c2C1 53192,N1(C(CCC=C)=O)CCC2CCCN(C(=O)CSCc3ccccc3)C2C1 53193,Cn1cc(C2CC(C(N3CCC(N4CCOC4=O)CC3)=O)C2)c(C2CC2)n1 53194,N1(C(CSS(C)(=O)=O)=O)CCCOC(CNC(=O)CC2CCCCO2)C1 53195,N1(C(CC(C(C)C)C)=O)CC2OCC(NC(C3(CCN(C)C)CC3)=O)C2C1 53196,c1(C(=O)NCC2(O)CC(NC(C3CC(F)(CO)C3)=O)C2)cc2ccccc2o1 53197,Cn1cc(C(=O)NCC23CC2CN(C(=O)CSCC2CCCO2)C3)c(O)nc1=O 53198,N1(C(c2cc(C)nn2C)=O)CCn2c(C(N3CCN(C)CC3)=O)cnc2C1C 53199,C(=O)(C(CCC)=CCCCC1CC1)NCC(CNC(C1(C=C)CC1)=O)F 53200,c1(CSCCC)ccc(C(=O)N(C)CC2(CNC(=O)C(CC)N(C)C)CC2)o1 53201,c1(CC2CCN(C(c3c(CN)occ3)=O)C2)ccc(Cl)cc1 53202,c1(C(=O)NCC2(CNC(CCN(C(CCC)C)C)=O)CC2)csc(Cl)c1Cl 53203,Cc1nn2c(C(=O)NCCCCNC(=O)C(C)C(C)C)c(C)nc2s1 53204,Cc1cc(=NC(=O)Cc2csc(=NCc3ccc(I)c(O)c3)[nH]2)[nH][nH]1 53205,N1(C(C2(COC)CN(C(C3(C)CCCCC3)=O)C2)=O)CCCC(C)(CCl)CC1 53206,c1(C(N2CCC(NC(C3CCCC34CC4)=O)(CF)C2)=O)cc2ccccc2cn1 53207,c1(NC(C(c2ccccc2)NC(C2CC(=O)NCC2)=O)=O)cccc2c1CCO2 53208,C1(CNC(CCCCN(C)C(c2ccn(C)c2)=O)=O)CCCC(C)(C)C1 53209,C1(OC)(OC)CC2(CC(NC(=O)NCCc3ccccc3)C2)C1.C1CCCN1 53210,CC(CCNC(C1CCC(C(N)=O)CC1)=O)CCNC(=O)C(c1ccnn1C)C 53211,C(C)(C)(CC(=O)NCCN(CCNc1cn(C2CCOC2)nn1)C1CC1)OCC 53212,c1(C(=O)NCc2nc(CNC(C3C(C)(C)C3)=O)sc2)cc(S(N)(=O)=O)ccn1 53213,C1(NC(C2(C#C)CN(C(=O)C(C)C#N)C2)=O)CCOCC12CCC2 53214,C1(C(=O)NCC(N(C(c2cnc(C(C)C)s2)=O)C)C2CC2)CCC(=O)N(C)C1 53215,N1(C(c2cn(CC)nc2)=O)CCC(C(=O)NCCCC2CCCCC2)C12CCC2 53216,N1(C(c2c(C)c[nH]c2)=O)CC(C)N(C(=O)C=CC(=O)N)CC1C.CC=CC 53217,c1(C(C)=O)ccc(C(N2CC(NC(c3c[nH]nc3OC)=O)CC2CO)=O)cc1C 53218,N1(c2cc(OC)ncn2)CCC2CC(CNC(c3ccc[nH]3)=O)CCC2C1 53219,O=C1CC2CC(C(N3CCC(C(=O)NC4(c5nc[nH]n5)CCC4)C(O)C3)=O)C1O2 53220,CC1CN(C(=O)CC(CC2CC2)NC(=O)C(C)(C)C(C)(C)C)Cc2c[nH]nc21 53221,CCCC(C)CC(=O)N1CCCC(CNC(c2ccc(-c3cc[nH]n3)s2)=O)CC1 53222,Cn1c(O)nc2c(N3CCN(CCC(F)(F)C(F)(F)F)CC3)ncnc12 53223,c1(C(N2CC(COC)(CNC(=O)C(F)(F)C3(O)CCC3)C2)=O)ccnc(C)c1O 53224,C1(NC(C(C)n2ccnn2)=O)CCC(C)(NC(C2COCCOC2)=O)CC1 53225,C1(CC)CCN(C(=O)C(F)F)C(C(=O)NCC2(C)CCCOC2)C1 53226,N1(C(c2c(C)ocn2)=O)CCN(C(=O)CNC(c2ncn(C)n2)=O)CC1 53227,c1(CC)cc(NC2CC(NC(=O)CCC(C)C)C2(C)C)ncn1 53228,C(=O)(C(O)C(F)(F)F)N1CC(N(C)C)C(NC(=O)CC(=O)NCC2CC2)C1 53229,c1(C(N2C(CNC(=O)C(O)C3CC3)CC(O)C2)=O)cnn2c1OCCC2 53230,C1(C(=O)OCC2N(CCC(C)C)CCC2)CCN(C(C2CCCO2)=O)CC1 53231,N1(C(c2cnc(CCC)s2)=O)CCCC(N(C)C(c2ccn(C(C)C)n2)=O)CC1 53232,C12(C(=O)NC3CC(NC(c4c(Cl)ccc(C)n4)=O)C3)C3C4C1C1C2C3C41C(N)=O 53233,N1(C(C(C)C2CCCC2)=O)CC2CCC1C2NC(c1ccc(Cl)c(O)c1)=O 53234,Cc1ccc(C=CC(=O)NC2CCN(C(C3CS(=O)(=O)CCO3)=O)CC2F)nc1 53235,c1(OCC(N2CCNCC2)=O)nccnc1C(=O)Nc1cccnc1 53236,C=CCCCC(C(=O)N1CCn2ncnc2C1)NC(c1cc[nH]c1C)=O 53237,Cc1c(CC(=O)NCCCNC(=O)CC2C=CCC2)cccc1[N+](=O)[O-] 53238,c1(CC)cc(C(=O)NCC(C(C)C)NC(=O)C(C2CCC2)OC)ncn1 53239,CC12CCN(C1)C2=O.C1(OCC(=O)NCC(F)(F)F)CC(=O)N1 53240,C1(OC)CC2(C1)CC(C(=O)NC1CC3CC1N(C(=O)C(O)CSC)C3)C2 53241,C1(NC(C2CCN(C(c3cn(CC=C)nc3)=O)C2)=O)CCN(C)CC1C#N 53242,C1(C(=O)NC(C)CC2CCOCC2)CCC(C)N1C(=O)CC1CC1C1CC1 53243,C(CCN=c1[nH]c(N2CCOC(CF)C2)nc2c1SCC2)OCC(C)C 53244,c1(CNC(C2CC(O)CN2C(c2nccnc2Br)=O)=O)ccc2cc[nH]c2c1 53245,Cc1cccc(C(=O)N(C)CC2CCCC2NC(C2(O)CCC(C)CC2)=O)c1N 53246,N1(c2ncc(OCC)cn2)CC(C(=O)O)C2(CCN2S(=O)(=O)CCBr)C1 53247,C1(NC(C2C(C)CCC2)=O)(CNC(C2CC(F)(F)C2)=O)CCOCC1 53248,C1(CNC(C2CN(C(=O)CO)CCO2)=O)COc2ccccc2O1 53249,C(c1cncnc1O)=CC(=O)NCCC(C)N(C)C(C1CCS1(=O)=O)=O 53250,C1(CC(C)NC(c2cn(C3CCOC3)nn2)=O)CCN(C(=O)CSC(F)F)CC1 53251,C1(C(=O)NCC(C)CC2CC2)CCC2CCC1N2C(=O)Cn1cnnc1O 53252,c1ccc2c(c1)CCC(n1nc(C3CCOC3)nc1-c1n[nH]c3c1CCC3)CC2 53253,CC(CC(=O)NOCc1ccccc1)C1CC1.C(=O)(C(F)(F)CO)O 53254,C(=O)(CC(C(F)(F)F)N(C)CC)NC1CN(C(C2(CC#C)CCCCO2)=O)CC1C 53255,N1(C(C2(CC#C)CCCCO2)=O)CCC(Nc2cc(F)ncn2)C(F)(F)CC1 53256,C(=O)(C1=CC2CCCC12)N(C1CCN(C(c2c(O)cccc2O)=O)C1)CC 53257,N1(C(CC2CN(C)C2)=O)CCCNC(=O)C1Cc1ccccc1 53258,C1(NC(C2CC3CC2C2CC32)=O)CCC2CN(C(=O)C=Cc3cscn3)CC2C1 53259,N1(C(C(CC2CCC2)NC(Cc2cccc(C#C)c2)=O)=O)CC(F)(F)CCC1C 53260,c1(OCCC)ccc(NC(=O)NCCOC2CC2(F)F)cc1OC 53261,Cc1sc2ncnc(N3CCC4CCC(NC(C5CCC(C)C5)=O)C3C4)c2c1C 53262,c1(C(N2CCC(CNC(CC(C)OC)=O)CC2)=O)ccc2c(c1)CC(C)(C)C2 53263,c1(CNC(=O)CCN2CCOC2=O)ccc(-c2ccccn2)cn1 53264,C=CC(F)(F)C(=O)N1CC2C(n3cc(-c4cc(C)nn4C)nn3)C2C1 53265,N1(C(c2cc(C(C)C)no2)=O)CCCC(NC(c2ccnc(Cl)c2O)=O)C1C 53266,C#CC1(CC)COCCN1C(c1nc(CO)cs1)C(=O)NC1CC(F)(F)C1 53267,C1(C(N2CCSCC2C2CCC2)C(=O)NC2(C)CC2)CCOC2(CCOCC2)C1 53268,N1(C(CC(CC)O)=O)CC(C)CN(C(c2[nH]cnc2C)=O)CC1C 53269,Cc1c[nH]c(=NCCC(C)NC(C2(C)CCCC2)=O)nc1C 53270,C1(C(=O)NCC(CN(C(=O)C(C)(C)N2CCCC2)C)(C)C)CCCCC1C(N)=O 53271,c1(CN(C(=O)CN(C2CCSC2)C)C)ccc(CNC(=O)CC2CCCO2)cc1 53272,CC1CN(C(c2cc(C3CCCC3)no2)=O)CCCN1C(C1CCCCC1O)=O 53273,Cc1sc(O)nc1C(N1CCCC(NC(c2cnc(Br)s2)=O)C1)=O 53274,C(=O)(CCCCC(N)=O)NC(C1CCN(C(c2cc(Cl)c[nH]2)=O)CC1)C(C)C 53275,N1(C(C2CC(C)(C)C2)=O)CC2CCCC(NC(c3nc(Cl)c(Cl)s3)=O)C2C1 53276,C1(C(N(C)CCNC(c2cccc(=O)o2)=O)=O)CC(C)(C)OC1(C)C 53277,C(=O)(C(C)(C)S(C)(=O)=O)NC1CN(C(c2c(OC)c(F)ccc2)=O)CC(C)C1 53278,CC(C)CCC(=O)NCCC1(CNC(C2(C(=O)N(C)C)CC2)=O)CC1.C12CC1C2 53279,C1(C#N)(C(CN2CCCC(C(N3CCOCC3)CNC(C)=O)C2)=O)CC12CCC2 53280,N1(C(Cc2n(C)cnn2)=O)CCN(C(=O)CCc2cccc(F)c2Br)C2CC12 53281,C1(C(=O)NCC2(CNC(CC(C)C)=O)CC2)CC(C)CC(C)(C)C1 53282,N#Cc1ccc(=NC2CCCN(C(c3cc4ncccc4[nH]3)=O)C2)[nH]n1 53283,C(CN=C(NCc1cc(Cl)ccc1Br)N1CCC(C2CCOC2)C1)N(CC)CC 53284,N1(C(CC(CC)SC)=O)CCC2(C=C(C(=O)N3CCN4CCCCC4C3)C2)C1 53285,c1(CC(N2CC(N(C(=O)CC(C)(C)F)C)C2)=O)noc2ccc(O)cc12 53286,Nc1c(C(N2CC(O)CCC2C(=O)NCc2ccc(F)cc2)=O)cccc1F 53287,C1(C(=O)N(CC(C)(C)CNC(C2(COCC)CC2CC)=O)C)(OC)CS(=O)(=O)C1 53288,c1(CC)cc(N)c(C(N2CCCC(C)CC2)=O)cc1F 53289,c1(C(=O)NCC2(O)CN(C(C(CC)C(C)O)=O)C2)cnc2c(F)cccn12 53290,CC1(C)CCCCC1n1nc(-c2ccc(Cl)nc2)nc1C1CCCC12CC2 53291,c1(NC(C)=O)ccc(C(=O)NC2(C)CCN(C(C34CCC3C4)=O)CC2)cc1Cl 53292,C1(C(N(C2CCN(C(=O)Cn3nnc(C)n3)CC2)CCC)=O)CN(C)CCO1 53293,c1(C(N2C(C(C)NC(C3ON=C(C)C3)=O)CCC2)=O)cc2cccnc2s1 53294,c1(CC)ncc(C(=O)NCCC2COCCN2C(=O)C(O)CCSC)c(O)n1 53295,Cc1nc(N2CC(NCc3ccc(F)c(C)c3)C3(CC3)C2)c2c[nH]nc2n1 53296,C1(NC(C=CC=CC)=O)CS(=O)(=O)CC1NC(C1(S(C)(=O)=O)CC1)=O 53297,C1(C(=O)NC(C)(CNC(=O)CCC2CC2)Cn2cccn2)CCC2CCC1O2 53298,C1(C(N2CCC(CNC(COCC(C)(C)C)=O)C2)=O)CCNC(=O)C1 53299,C(=O)(C(CC(C)C)OC)NC1CC(C(=O)NCC(=O)OCC#C)C1(C)C 53300,CCCCC(=O)C(=O)N1CC(C)CC1C(N1CCCC(CN(C)C)C1)=O 53301,C1(C(N(C)CC2CCCN2C(c2ccc(Cl)o2)=O)=O)CC2CC1C1CC21 53302,C1(CNC(C(C)C)=O)COCC2(CCN(C(C3(F)CCC3)=O)C2)O1 53303,CCCCCC(=O)N1CCC(F)(CNC(=O)C(C(C)C)c2cnn(C)c2)C1 53304,C(=O)(C1CCCc2cn(C)nc21)NC(C)CCC(C)(C)O 53305,C1(C2CCN(C(c3cncc(Cl)c3)=O)C2)(NC(C(Cc2c(C)nc[nH]2)O)=O)CC1 53306,C(=O)(CCC(C)(C)F)NC1C(C)CN(C(c2ccc(C(F)F)o2)=O)C1 53307,C1(CNC(c2n(C)cnc2)=O)CCC(F)(CNC(C2(C)CCCNC2=O)=O)CC1 53308,N1(C(C(CCC)C(C)C)=O)CCC2(CC1)COC(CNC(c1cscn1)=O)C2 53309,c1(OC)cc(CC(C(=O)N(C)C)NC(N2CCCC23CC3)=O)cc(F)c1F 53310,CC(C)CCC(O)C(=O)NC1CCN(C(=O)C2=COCC2)CC(O)C1 53311,N1(C(c2c(C)occ2)=O)CCCC2(NC(c3ccccc3Br)=O)CC2C1 53312,Cc1oc(Br)cc1C(N1CC(F)(CNC(C2CC23CC(O)C3)=O)C1)=O 53313,N1(C(C=COCC)=O)CCOCC1CNC(=O)C(C)=C(C)C(c1ccccc1)=O 53314,Cc1c(F)ccc(C(N2CCOCC2)C(=O)N(C2CC2)Cc2ccccc2)c1Cl 53315,c1(C(=O)NC(CN(C(C(CC=C)CC)=O)C)CC)cc(C)nc2[nH]c(=N)sc12 53316,C1(CC(N2CCCC(C)C2CNC(=O)C=C2CCCC2)=O)Cc2ccccc2N1 53317,N1(C(c2cn(C)nc2C(F)(F)F)=O)CC2CCC(C1)N2C(=O)CC1CCC1 53318,C1(C(N2CC(C(N)=O)(CNC(C3(CO)CCCC3)=O)C2)=O)CC2CCC1C2 53319,N1(C(c2scc(COC)c2)=O)CCOCC1Cc1cn(-c2cccc(C)n2)nn1 53320,Cc1coc(C)c1C(=O)NCC(C)CN(C(=O)CSCc1csc(=N)[nH]1)C 53321,n1(CC)nc(C)cc1C(=O)NCC1CCC1NC(=O)CN1CCCCC1C 53322,CCC(O)C(C)C(=O)NCC(C)(C(C)C)NC(=O)Cc1ccc(Cl)nc1 53323,c1(CC)nccnc1CNC(=O)C(C)(CSC)NC(=O)C=CC1(C)COC1 53324,Cc1cn2c(n1)C(C)CC(C(=O)NC1CCC1NC(=O)CCC(C)(C)C)C2 53325,N1(C(C(CC=C)CNC(=O)C=Cc2cncn2C)=O)CC2CCC(CC2)C1 53326,c1(C(N2CCC(C)(NC(c3n(C)c(S)nc3)=O)C2)=O)nc2c(s1)COCC2 53327,C(=O)(CCC(F)(F)CN=[N+]=[N-])NC1CC(C)(CNC(C=CCOCCOC)=O)C1 53328,CC1(C)CCN(C(C2CCCC(=O)N2)=O)C1CNC(C1(C(N)=O)CC1)=O 53329,C(=O)(CC1CCCc2ccccc21)NC1CC(CNC(C2(C)CC=CCC2)=O)C1 53330,C(=O)(C1=COCCC1)NCCC1CCN(C(C(C(C)C)OCC(C)C)=O)C1 53331,N1(C(C(CC)=CC)=O)CC(NC(=O)CC(C)n2ccc(C)n2)C(C)C1 53332,n1(CC)nc2c(c1C(N1CC3CC1CN3C(=O)C(F)CCC(C)(C)C)=O)CCCC2 53333,CN1CCCC1(C)CNC(=O)Nc1nc(-c2ccncc2)cs1 53334,C1(OC)CC(C(=O)NCC(C)(C)CN(C)C(C2CCN(C)CC2)=O)C12CCC2 53335,C(=O)(C1=CCCN(C(c2ncccc2F)=O)C1)NC(c1ccc(O)nc1)C 53336,C1(C(=O)NC(c2ncc[nH]2)C)CN(C(=O)C(c2ccn(C)n2)C)CC12CCC2 53337,c1(OC)cc(NC(=O)C(C)N(C(=O)CC(C)n2ccnc2)C)ccc1F 53338,c1(C(N2CC(C(C)NC(CCSCCCC)=O)OCC2)=O)cccc(C)c1Cl 53339,N1(C(C2C(CC(C)C)C2)=O)CC2CN(C(=O)C=CC3COC(C)(C)O3)CC2C1 53340,c1(N(CCC)CCNC(=O)CC2=NNC(=O)C2)cnc2cc(F)c(F)cc2n1 53341,n1(C(C(=O)N(CC(C)C)C(C)C2CC2)C)cc(C(C)N(C)C)nn1 53342,C1(OCCCC)CCN(c2nnc(-c3n[nH]c(=N)[nH]3)n2CC2CCC(F)C2)CC1 53343,C#CCC(C)(C)C(=O)NCC(CC=C)C(=O)NC(CC=C)C(=O)OC 53344,CC1=NN(C)C(=O)C1CC(=O)NCC1(CNC(=O)COC(C)C2CC2)CC1 53345,C1(C(N(C(C)CNC(=O)CC2COCCO2)C)=O)CCCCN1C 53346,N1(C(C2C(COC)C2)=O)CCC(C(C(C)C)NC(C2C(C(F)F)C2(C)C)=O)CC1 53347,C1(NC)CC2(C1)CC(C(N(Cc1cccnc1)Cc1ccc(C(=O)O)cc1)=O)C2 53348,c1(OC)ccc(C(N2CCN(C(=O)CNC(C)=O)CC2)C(=O)NCCC#N)nc1 53349,C1(C(=O)NCCc2cn(C(C)(C)OC)nn2)CCCC(=O)C1 53350,c1(C(=O)OC)cc(C(=O)NC2CCC2NC(=O)COC2CC=CC2)ccc1F 53351,N1(C(C(CC)COC)=O)CCCC2(CCCN2C(=O)C2=C(Cl)CCCC2)C1 53352,c1(NC(C2CCN(C(CCN(C)CC)=O)C2C)=O)cc(C)cnc1O 53353,C1(CCC)CC(C(=O)NC2CN(C(=O)Cc3cnco3)CC2C)CCO1 53354,CC#CCCC(=O)NC(CC1CC1)C(=O)NCCN1CCCC1C 53355,c1(C(N(CCNC(c2cnc(Cl)s2)=O)CC2CC2)=O)nnc2ccccc2n1 53356,N1(C(C(N2CC(C)C2)C)=O)CCCCC1CC(=O)NCc1cnc[nH]1 53357,Cc1cc2nc(C(N3CCC(C(C)NC(c4cscc4C)=O)C3)=O)cn2cc1C 53358,N1(C(CC2N(C(c3c(C)nc(C)[nH]3)=O)CCC2)=O)CC=C(c2ccccc2)CC1 53359,C(=O)(C1=C(C)OCCC1)NC1C(NC(c2nc(OC)c(F)cn2)=O)CCC1 53360,c1(C(=O)NC2CCC(N(C)C)C2)cncc(OC2CCCCC2)c1 53361,Cc1ccnc2sc(-c3nc(CCCC#N)nn3CC3CC3C)c(C)c12 53362,c1(OC)ccc(CN2CCC(C(C)CO)CC2)cc1-c1c(C(=O)O)nn(C)c1O 53363,Cc1nnc(O)c(C(=O)NCC2C3CCCC2N(C(=O)Cc2ccco2)C3)c1C 53364,N1(C(C2=NOC(C)C2)=O)C2CCC1CC(NC(=O)Cc1ccc([N+](=O)[O-])cc1)C2 53365,c1(C(CC)OC(=O)CC2ON=C(C)C2C)ccc(Cn2cccn2)cc1 53366,C1(C(N(CCCOC)CCO)=O)CCC(C)(C)N(C(=O)C(CO)C(F)(F)F)C1 53367,N1(C(C(COC)N(C)C)=O)CCCCC1C(=O)Nc1cccc(C)n1 53368,Cc1cc(C(N2CCOCC2C(=O)NCc2[nH]ccc(=O)c2O)=O)ccc1F 53369,C1(NC(C(CC)N(C)C)=O)CCC12CCN(C(c1oc(CO)cc1C)=O)CC2 53370,N1(C(C2N(C(C(c3ccc(OC)cc3)C)=O)CC=C2)=O)CCCC2(COC2)C1 53371,N1(C(C(=O)NCCC)CC2CC2(Cl)Cl)CCOCC1(C)Cc1ccccc1 53372,C1(CC)CN(C(=O)CN2CCC(F)CC2)CC1C(=O)N(C)CCSC 53373,c1(C(=O)NCCCC(C)NC(C2(F)CC=CC2)=O)nn(C)c2c1CS(=O)(=O)CC2 53374,C1(C(=O)Nc2nc(C)ncc2Br)(OC)CCN(C(C2CC2F)=O)CC1 53375,N1(C(C2C(=C)C2)=O)CCN(C(C2C(C(C)=O)C2(C)C)=O)C(C2CCCC2)C1 53376,C1(N(C(C(C)OCC2CCCO2)=O)CC2CC2)CCN(C(=O)CCc2ccc[nH]2)C1 53377,C12(C3CC3)CCN(C1)C(=O)CN2.c1(CNC(c2cccnc2)=O)ccc(C2CC2)o1 53378,c1(COCC)cn(CCCC(=O)NCc2ccsc2C(=O)O)nn1 53379,C(C(CC(=O)NCCC1CCC(C)(C)O1)NC(=O)C(O)CCSC)OC 53380,N1(C(C2=NNC(=O)C2)=O)CC2CC1CN(C(c1nccn3nccc13)=O)C2 53381,C(=O)(CCC(C)N(C)C)NCC(=CC(=O)NCC1(COC)CCCO1)C 53382,c1(CC(C(=O)OC)NC2(C)CCC(=O)N(C)C2)ccc2c(c1)CC(C)O2 53383,C(=O)(CCP(C)(C)=O)N1CCC(N(CC#C)C(c2nc(C)oc2C)=O)C1 53384,CC1CCC2(CC1)CCN2C(=O)CCCCCCn1cc(-c2ccc(Cl)cc2)nn1 53385,C(C(=O)N1CCN(C(C2CCCCN2CC(F)F)=O)CC1C)(C(C)(C)C)SC 53386,Cn1ccc(C(=O)NCC2CCCN(C(C3(C(F)F)CC3(F)F)=O)C2)cc1=O 53387,c1(C(C)(C(=O)NCC(CNC(=O)CCCC2CC2)CO)N(C)C)ccc(F)cc1 53388,N1(C(c2cc(N)c(Cl)cn2)=O)CCOC2CN(C(=O)CC3C=CCC3)CC12 53389,C(C(CCO)NC(C1=NOCC1)c1nnnn1CC1CC1)OC(C)(C)C 53390,n1(CC2CC(=O)C2)cc(C(=O)NCC2CC2NC(c2cc(C(F)F)c[nH]2)=O)cn1 53391,N1(C(CCC2(C)CC2)C(=O)NCC2CC2)CCC(S(=O)(=O)C(C)(C)C)C1 53392,C1(CNC(=O)Cn2ccc(C3CC3)n2)CC2(CCC2)CN1C(=O)CCSC1CC1 53393,N1(C(Cn2cc(C(=O)NC)nn2)=O)CC2ON=C(CNC(=O)C=CC(C)C)C2C1 53394,c1(C(=O)NCC2C(NC(c3cnc4[nH]cncc3-4)=O)C2)ccc(Cl)c(F)c1F 53395,N1(C(C=CCCC)=O)CC2CC(C(N3CCC(CO)C(C)C3)=O)C(C2)C1 53396,Cc1ccccc1C=CC(=O)NC1CC2(C1)CC2NC(C1CCC(=O)N1C)=O 53397,N1(C(COCC=C)=O)CC2CC(NC(=O)CC(C)(C)CC)CC1C2 53398,CCC(CC(=O)NC(C)CCCNC(c1nc(C(C)C)oc1C)=O)C1CC1 53399,c1(C(CC)C)ccccc1OCC(=O)NCc1ccn(C(F)(F)F)n1 53400,C(=O)(C(O)CC(F)(F)F)N(CCC(=O)N1CC(N2CC(O)C2)C1)CC1CC1 53401,Cc1cc(Oc2ccccc2)c(CC(=O)NNC(=O)c2cc(C)oc2C)cc1Cl 53402,C1CCC2C(N3CCC(OCC4CCCO4)C3)C2CC1 53403,CCC(CC)N(C(=O)COC(C1CC1C1CCCO1)=O)CC 53404,C1(C(N2CC(OCCOC)C2)=O)CCC(CNC(=O)CCCF)O1 53405,C1(CN(C(CC(CC)C2CCC2)=O)C)CCCN(C)C1c1ccnn1C 53406,N1(C(C2CNC(=O)N2)=O)CC(NC(c2ccoc2Br)=O)C2(CCC2)C1 53407,c1(C(=O)NCC(CNC(CC(C)O)=O)F)c(Br)ccc2n[nH]cc12 53408,C1(C(=O)NCC(C2CCC2)OCC)(CO)CCN(C(C2CCN(C)C2)=O)C1 53409,N1(C(C2C3CN(C(C4C(OC)CCCC4)=O)CC32)=O)CC2CC2C2CC12 53410,c1(C(=O)NCCCN(C)C(c2cnc3ccoc3c2)=O)cncc(P(C)(C)=O)c1 53411,C(C1=NOC2CCCC12)NC(CCOCCCNC(CNS(N)(=O)=O)=O)=O 53412,C1(O)(CC(N2CC(CCNC(=O)C(O)c3ccco3)C2)=O)CCCOC1 53413,c1(C(=O)NCC2N(C(CN3CCN(C)CC3)=O)CCC2)cncc(C#N)n1 53414,c1(OCCNC(N2CC(C)(C#N)C2)=O)ccc(N=[N+]=[N-])cc1 53415,C1(N(C(c2cscc2Br)C(=O)NC(C(=O)OC)C)C)CCC2COC1O2 53416,c1(C(=O)NCC2(NC(C(CC)F)=O)CCC2)ncn2ccc(C)cc12 53417,CCC(C)CCC(O)CC(=O)N1CCCC1C1CCN(C(=O)CCCOCC=C)C1 53418,C1(CNC(C2C(C(N)=O)C2)=O)C2CC1N(C(C1CCCC1F)=O)C2 53419,c1(C(=O)NC2C(CNC(Cc3n(C)nc(CC)c3Cl)=O)C2)nc2c(s1)COCC2 53420,C1(NC(=O)CN(C(=O)C2CC2)C2CC2)C2CN(C(C3(n4cncn4)CC3)=O)CC12 53421,c1(C(N(CCNC(=O)OC)CC)=O)cc2sc(CC3CC3)cc2o1.C1CC12CC2 53422,CCC(C)(C)C(=O)C(=O)N1CCC(C(=O)NOCc2ccccc2F)C(O)C1 53423,c1(C(N2CC(NC(c3c(C)onc3CO)=O)C2)=O)ccc(S(=O)(=O)C(F)F)cc1 53424,c1(CN2CCN(Cc3ccc(C(CC)N(C)C)cc3)CC2)cc(Br)ccc1Cl 53425,C(=O)(CC(N)C(=O)NCCC(C1CCC(O)C1O)=O)OC 53426,N#Cc1ccc(C(=O)Nc2cccc(NC(=O)CC3CC4CC4C3)c2)cn1 53427,c1(C2CN(NC(C3C(C)(C)C3)=O)C2)ocnc1-c1cn(CCC=CCO)nn1 53428,CC1(C#CC(=O)N2CCC(CO)CC2)CN(C(C2COCCO2)=O)C1 53429,c1(C(N(C2CCCCCC2)CCNC(CCSC)=O)=O)cc(F)c(F)c(Cl)c1F 53430,N1(C(C(C)NC(CC)=O)=O)CCCN(C(c2cnc(C(C)C)nc2)=O)CC1C 53431,n1(CC)ccnc1C=CC(N1CCOC(CCNC(C2CCS2(=O)=O)=O)C1)=O 53432,C(=O)(C(F)C1=CCCCC1)NCC(C1CCCC1)NC(c1c(CC)n[nH]c1)=O 53433,c1(CNC(CSC)=O)cc(C(=O)NC(C)CC(N)=O)no1 53434,N1(C(C(C)SCC)=O)CCCC(C)(CNC(=O)CCc2cc(C)nc(C)c2)C1 53435,C1(NC(CCN(CCCO)C(C2(OC(C)=O)CC2)=O)=O)CCCC2(C1)N=N2 53436,C1(NC(C(C=C)C)=O)CCCCC1NC(=O)CCc1cc(C)no1 53437,c1(CNC(=O)Cc2ccon2)nc2c(s1)CN(C(=O)C(O)(C1CC1)C1CC1)CC2 53438,CC(C)CCC(O)C(=O)NC(Cc1ccoc1)C(=O)NC(C1CCCCC1)C 53439,c1(C(=O)NC(CNC(C2(C)CC2Br)=O)CO)cncc2sccc12 53440,O=C(N=c1cc[nH]cc1F)C12CCN(C(c3ccc(Cl)c([N+](=O)[O-])c3)=O)CC1C2 53441,N1(C(C(=O)NCCc2ccc(OC)cn2)=O)CCC(C)C(C)C1 53442,c1(CN(CC(C)(C)SC)C)c[nH]c2cccc(Br)c12 53443,c1(C(N(C2CCC(NC(c3ccc(F)o3)=O)C2)C)=O)csc(Br)c1 53444,C1(CNC(C(c2cncnc2)C)=O)CC2CCC1N2C(c1ncccc1Cl)=O 53445,C(C(C)(C)CC(=O)N1CCCC1)c1nc(-c2c(C)oc(C(C)(C)C)c2)on1 53446,CCCC(C)(C)CC(=O)N1CCC(NC(=O)CS(=O)(=O)CCO)C(C)C1 53447,c1(C(N2CCN(C)CC2CNC(c2ccnnc2O)=O)=O)cc2c(o1)CCCC2 53448,C1(NC(c2cc(N)sc2)=O)CC2(NC(c3cc(-c4ccco4)no3)=O)COC1C2 53449,CON=C(C(=O)N(C(CNC(=O)C(C)(C)C1CCCO1)C1CC1)C)c1ccco1 53450,N1(C(C2CN(C(C3CCN(C)C3)=O)CC(F)(F)C2)=O)CCC2(CC1)CC(=O)N2 53451,c1(C(=O)NC2C(C)N(c3cncc(Cl)n3)CCC2)ccc2c(c1)ncn2C 53452,N1(C(C(C2CCN(C(CS(CC)=O)=O)CC2)C)=O)CCc2nn[nH]c2C1 53453,c1(NC)cccc(C(N2CC(F)CC2CNC(c2cnn(C(C)C)c2)=O)=O)n1 53454,N1(C(c2c(CC)nc(C)o2)=O)CC(NC(=O)C(C(C)C)C2CCC2)CC(F)C1 53455,c1(C(N(C(C)C2CC2)C)=O)n[nH]c2c1CN(C(C1(C)CCC(=O)N1)=O)C2 53456,c1(C(=O)NC(CN(C(CCCOCCC)=O)CC)C)cc(Cl)ccn1 53457,c1(C(C(=O)NCCCN(C(C23CCC(CC2)O3)=O)CC)=O)cc(F)cc(Cl)c1 53458,N1(C(c2c(C)n(CCO)cc2)=O)CCC(NC(c2cc(C3CC3)no2)=O)C12CC2 53459,C1(NC(C(CSC)O)=O)CCCC(C(=O)N(C2C3CCCC23)C)CC1 53460,N1(C(C(C)CO)=O)CCC(CCC(=O)NC2CCOC2)CC1 53461,c1(OC)ccc(CC(=O)NC(C)(C)CNC(c2cc(CN(C)C)on2)=O)c(C)c1 53462,c1(C(=O)NCC(CC)(C)NC(C2CC2F)=O)ccc(F)cc1OC 53463,C1(C(=O)NCCC(CCC)O)CCCCN(C(c2cnn(C)c2OC)=O)C1 53464,C=CC(C)C(=O)N(CCC(=O)N(C1CCC1)CCO)C 53465,C1(C(=O)NCc2cn(C3CCN(C(CC)=O)CC3)nn2)CCS(=O)(=O)C1(C)C 53466,N1(C(C(C)(C)CC2CC2)=O)CCC2(CCN(C(c3csc(CO)n3)=O)C2)C1 53467,Cn1ncc(NC(C23CC(CN2C(C2CCCC(F)C2)=O)C3)=O)c1C(N)=O 53468,Fc1cncc(CCc2nc(-c3ccccc3)nn2C2(c3cccs3)CC2)c1 53469,C(N=c1[nH]c(=NC2CCOCC2)[nH]c2c1CCC2)C1(S(C)(=O)=O)CC1C(=O)O 53470,C1(C(=O)NCC(CC)CCO)CN(C(c2ncn3c2CCC3)=O)CC(C)O1 53471,C1(CNC(C2(OC)CCC2)=O)CC2(CCC2)CN1C(=O)CCC1CC(F)(F)C1 53472,C1(NC(c2n(C(CC)C)ncc2)=O)(CO)CCCN(Cc2ccc(Br)s2)C1 53473,C(=O)(C(C)P(C)(C)=O)N1CCC1.c1(C(=O)OCC)occc1Cn1cc(Br)cn1 53474,C1(C)(CC(=O)NCc2snc(C)n2)CCN(C(c2sccc2F)=O)C1 53475,N1(C(CCC2C(C)C2)=O)CCOCC1CCNC(c1cc(C2CCCC2)no1)=O 53476,C=CC1(CC(=O)NCC(=C)F)CN(C(c2cc(OC)ns2)=O)C1 53477,c1(-c2ccc(C(=O)NC3C(N)CC3)s2)cc(OC(F)(F)F)cc(F)c1 53478,n1(CC)nc(C(=O)NCCN(C)C(c2csc(COC)n2)=O)c(C)n1 53479,CC(C)CC(O)C(=O)NCCCOC1CCN(C(=O)CSC(F)F)C1 53480,c1(OC)ncnc(N2CCOC(C(C)NC(c3cnccn3)=O)C2)c1OC 53481,N1(C(C(C)(F)F)=O)CC2CCN(C(c3ccnc(C(C)(F)F)c3)=O)C(C2)C1 53482,C(=O)(C(C)(C)S(C)(=O)=O)NCC1C(C)CCN1C(=O)Cn1ccc(C(F)F)n1 53483,N1(C(=O)NCC(C(C)C)C)c2ccc(Cl)cc2OCC1C 53484,N1(C(C2(CCC=C)CN(C(c3cccc(C)c3O)=O)C2)=O)CC2CCCC2C1 53485,C12(C(=O)NCC3(NC(c4ncccn4)=O)CCCC3)COCC1CS(=O)(=O)C2 53486,C=CC(CCC)CC(=O)N(C)CC1CN(C(c2ccccc2)=O)CCO1 53487,CC1(NC(=O)COCc2cc(CO)cs2)CCN(C(=O)CCC2CCOCC2)C1 53488,C=CCC(C)(CC)C(=O)N1CCC(NC(c2ccnc(C(F)(F)F)n2)=O)CC1 53489,C1(C#N)(C(N2CC(NC(c3ccc(OC)s3)=O)C(C)C2)=O)CCSCC1 53490,c1(C(N2CCC(CNC(=O)COCC3CCCO3)C2)=O)cccc2[nH]cc(Cl)c12 53491,C=CCC(C)(C)CC(=O)NC(CCF)C(=O)N(CCC)CC 53492,C1(C(=O)NCC2(C)CC(C)C2)CC1C1CN(C(C2CCCC(C#N)C2)=O)C1 53493,c1(C(=O)NC2(C)CN(C(C(CCC)CC)=O)C2)cc2c(C)cccc2[nH]1 53494,N1(C(CC(C)(C)C)=O)CC(NC(=O)CCc2nc3ccccc3s2)C(C2CC2)C1 53495,N1(C(C(C)N=[N+]=[N-])=O)CC2COCC2(C(N2CCSC(C)C2)=O)C1 53496,C(=O)(C1OCCc2ccccc21)NC(CCN(C(c1c(COC)nn[nH]1)=O)C)C 53497,CC1(C#CC(=O)N2CCCC2C2CCN(C(c3ccc(C4CC4)s3)=O)CC2)CC1 53498,C#CC1(C(=O)Nc2ccc(SC)cc2)CCN(C(=O)CSc2nncn2C)CC1 53499,N1(C(CN(C2CC2)CC)=O)CC=CC(NC(c2cccc(C(C)(C)C)n2)=O)C1 53500,CCCCCCC(CNC(c1nc(C)c(C)nc1C)c1nnnn1C)CC 53501,CN1CCN(C(=O)CCc2nccs2)C(C(=O)NC2C3CCC(F)(F)C23)C1 53502,c1(NC(c2nc(C)on2)(C)C2CC2)cc(-c2ccc(Cl)cc2)ncn1 53503,c1(C(=O)NCC2CCCCN2C(=O)CCN2CCOC2=O)n[nH]c2c1CC1CC21 53504,C12CN(CCCO1)C2=O.C(C(O)C(=O)Nc1ccccc1)NC(=O)OC(C)(C)C 53505,c1(C(=O)NC23CC(NC(c4ccnc(F)c4Cl)=O)(C2)C3)cc2cc[nH]c2cc1F 53506,N1(C(C(C=CC)O)=O)CC2(CC(NC(c3c(C)cc(C)nc3S)=O)CO2)C1 53507,c1(CNC(c2nnc(C)n2C)c2n(CCOC)nnn2)cccc(Br)c1 53508,C(=O)(C(CCC(C)C)NC(=O)C(=O)NCC1CC1)NC1C(CC=C)COC1 53509,C1(NC(c2ncn(C)n2)=O)CCCC12CN(C(C1CCCOCC1)=O)C2 53510,Cc1cncc(CCC(=O)NC2C=CCN(C(c3sccc3CC#N)=O)C2)c1 53511,C(C(C(F)(F)F)CCn1cncn1)NC(=O)CCCn1cc(-c2cccs2)nn1 53512,N1(C(C2C3CN(C)CC32)=O)CCC(C(N2CCC(F)(F)CC2)=O)C(C)(C)C1 53513,c1(C(=O)NCCCCn2cc(CNC(N)=O)nn2)cc(Br)sc1Cl 53514,Cc1cccc(C)c1NCC(N1CCCN(C(=O)CCC2CCC(C)O2)CC1)=O 53515,NC1CN(C(C2(Cc3ccc(F)cc3)CCCN2)=O)CCc2ccccc21 53516,C1(C(=O)NC2(CO)CCN(C(C=CC=CC)=O)C2)CCn2nccc2C1 53517,C1(OCC)(CNC(=O)C(=O)NC2CCC(C)S2)CCC(F)(F)CC1 53518,c1(C(=O)OCC(ONC(C(=O)OCC)=O)(C)C)csc(=NC2CC2)[nH]1 53519,c1(C(=O)NCCN(C)C(C2CCOC2C2CC2)=O)ccccc1OC(F)F 53520,CC(C)C#CC(=O)N1CCC(O)(CCNC(=O)C(C)CN2CCOCC2)C1 53521,C1(CCC(=O)NC(C(C)NC(CCCCCC)=O)CO)CCc2cnn(C)c2C1 53522,Cc1[nH]c2ccccc2c1C(N1CC(C)CN(C(=O)CCOC2CC2)C(C)C1)=O 53523,c1(C(=O)NCCCN(C(C2(n3nccn3)CC2)=O)CC)ccc[nH]1 53524,CCN=C(NCC1(O)CCCCC1(C)C)N1CCN(S(C)(=O)=O)CC1 53525,C(C(F)(F)C(=O)NC1CCC(NC(=O)C(c2cccc(Cl)c2)C)C1)OC 53526,CN=c1[nH]nc(CC(=O)NCC2(O)CCN(C(=O)Cn3ccccc3=O)C2)s1 53527,C1(CNC(c2cnc(C)o2)=O)CC(C)CCN1C(=O)C(Cc1ccsc1)NC=O 53528,N1(C(c2c(C)n(CC3CC3)cc2)=O)CCN(C(C2(NC(C)C)CC2)=O)CCC1C 53529,c1(CN2C(CNC(=O)C=CC(N3CCCC3)=O)CSCC2)c(Cl)ccc(F)c1F 53530,C(=O)(C(C)(C)S(=O)(=O)C1CC1)N(CCN(C(c1cccc(COC)c1)=O)C)C 53531,N1(C(C2C(C#N)C2)=O)CC2CC2(CNC(c2cn(CCO)nn2)=O)C1 53532,N1(C(C)=O)CC2(CCC(NC(c3c(Br)noc3C)=O)C2)C1 53533,C1=CC(=O)Nc2c(N)ccc1c2.C1(CC=C)C(OC(C)(C)C)CC1OC 53534,n1(CC(=O)NC(CN(C(C(C)OCCCCCC)=O)CC)CC)cccnc1=O 53535,c1(CC)nn(C)c(C(=O)NC(C)C(CO)NC(C2CC(C(C)C)C2)=O)c1Cl 53536,N1(C(=O)C(O)C(F)F)CCC2(CCCN2C(c2ccc(N3CCCC3)nc2)=O)C1 53537,c1(C(=O)NCCNC(C(CC)F)=O)cc2c(cn1)NC(=O)CO2 53538,N12CC(C(N)=O)(C1)COC2=O.c1(CC(=O)N(C(C)(C)C)CCO)cc[nH]c1 53539,c1(C(N(C2CC2)Cc2ccc(OC)c(F)c2)=O)n[nH]c2c1CC1CC21 53540,C1(O)(C(=O)NC2CN(C(C(COCC)N=[N+]=[N-])=O)CC2C)CCCC(C)CC1 53541,C1(O)(CNC(CC(C)c2ccncc2)=O)CCCN(C(C2(F)CCCCC2)=O)C1 53542,CN1CC=C(C(=O)NCc2ncc(C(N3CC(O)CC3C3CC3)=O)cn2)C1 53543,CC#CCC(C(=O)N1CC(N2CCOC2=O)C1)NC(c1c[nH]c(C)c1)=O 53544,C1(C(N(C2CCN(C(=O)C(C)N3CCCC3)CC2)CC#C)=O)CCC(F)CC1 53545,c1(C(=O)NC2CCN(C(=O)C3=CCCC3)C(C3CC3)C2)ccn2cccc2c1 53546,N1(C(c2c(CC)ccs2)=O)CC2CCC(CNC(c3cncnc3CC)=O)(C2)C1 53547,c1(SC)c(C(=O)NC23CC(NC(=O)COCCN(C)C)(C2)C3)cnn1C 53548,N1(C(C(CC(C)C)F)=O)CCc2sccc2C1CNC(=O)CC(C)(C)CC(F)F 53549,N1(C(C=CNS(N)(=O)=O)=O)CC2CCOCC2(NC(=O)C=Cc2cccnc2)C1 53550,CC(C(=O)NOCC(N1CC(CO)(CO)C1)=O)C1CCCC1 53551,C(=O)(C(CCCCC(=O)OC)N1CCCC(CCO)C1)NCCC 53552,Cc1ncc2c(n1)CCC(C(=O)NC1CN(C(=O)C#CC3(C)COC3)CC1C)C2 53553,N1(C(C2CCOC2)=O)CC2OCCN(C(c3cc(C4CCOCC4)[nH]n3)=O)C2C1 53554,C(=O)(CCN(C1CN(C(=O)C(C)OC2CCCC2)C1)CCCC)OCC 53555,c1(CC)nocc1C(=O)NCCN(C(=O)C(C)COC)C 53556,C(=O)(CC(C)(O)CCC)N(C1C(C)CCN(C(C(C=C)c2ccccc2)=O)C1)C 53557,c1(C(N2CCC(CN(C(CNC(C(CC)C)=O)=O)C)C2)=O)cccnc1C 53558,N1(C(=O)NCc2cnc3n2CCCCC3)CCCCC(C2CCOCC2)C1 53559,N1(C(C(C=C)O)=O)CCC(CO)C(NC(c2ccc(Br)c(C)c2)=O)C1 53560,c1(C(=O)NC2CC(F)(CNC(C(CC=C)CC)=O)C2)cc2nn[nH]c2cc1F 53561,Cc1ccc2c(c1)CCN(CCc1cc3cc(Cl)ccc3[nH]1)C2 53562,c1(COC(C(N(C)C(c2ccoc2)=O)C2CC2)=O)nc(O)c2ccccc2n1 53563,N1(CCNc2scc(-c3ccc(Br)cc3)n2)CCC2CCCC(C1)N2 53564,N1(C(c2ccc(SC)s2)=O)CC(NC(=O)CCSC(F)(F)F)C(C)C1 53565,c1(CC)[nH]nc(Cl)c1C(=O)NC1CC2C(NC(c3ncsc3C)=O)C2C1 53566,N1(C(C)=O)CCCCC1CC(=O)NC1(C)CC(NC(C2CCNC2=O)=O)C1 53567,Cc1cc(COC(=O)C(C)Oc2ccccc2C#N)cc(C)c1Br 53568,C(=O)(CCCC(=O)N(C)CC1COCCN1C(c1cncc(Cl)c1)=O)N(C)C 53569,c1(C(=O)NC(CNC(C=C(CCC)C)=O)CO)ccc(C(C)C)c(Cl)c1 53570,c1(C(N2CCN(CC)CC2(C)C)=O)c(OC)ccc(S(N)(=O)=O)c1OC 53571,c1(-c2cn(C3C(CC(C)C(=O)N4CCCC4)CC3)nn2)ncnc2ccc(Cl)cc12 53572,C#Cc1cc(F)c(C(=O)NC2CCN(C(C3CCC(C)(C)CC3)=O)C2)c(F)c1 53573,c1(C(=O)NC2C(NC(C=CC(C)(C)SC)=O)CCCC2)ncc(Br)cc1N 53574,Cc1ccc(-c2ccc(C(=O)NC(C)(C)CCNC(C3CCC(C)O3)=O)s2)s1 53575,CCCC(C#N)C(=O)NCC(CNC(c1cccc(Br)c1)=O)OC 53576,c1(OC)cc(NC(C2C3CC2N(Cc2cc(Cl)ccc2I)C3)=O)ccc1C 53577,c1(C(N2CCCC(C)C2CNC(=O)C(C)C2CCCO2)=O)cncc2[nH]ccc12 53578,c1(C(=O)NCC2CCCN2C(=O)CSc2nc[nH]n2)cccc(-c2nccs2)c1 53579,c1(C(N(CC)CC2CCCN2C(=O)CC(C)(C)O)=O)cc(Cl)cc(Cl)c1 53580,N1(C(CCCN(C(C)=O)C)=O)CCC(C)(C)C1C(=O)N(C1CC(O)C1)C 53581,C1(N(C(=O)CC2CSC2)CC)CCN(C(=O)C(C2CCOCC2)F)CC1 53582,C(CC(CC)C(=O)NC1CC(C)(NC(=O)C(CC)C(=O)OCC)C1)=CC 53583,c1(NC(CN(C(=O)CN2C(C)CCC2C)CCC)=O)ccc(F)c(O)c1 53584,C(=O)(CCCCCCC(=O)N1CCN(Cc2c(O)cccc2Br)C2CC12)OC 53585,Cc1cc(C(=O)NCCN(C(=O)C(O)CC(N)=O)C2CC2)cc(S(N)(=O)=O)c1C 53586,C(=O)(C(C(C)C)NC(=O)C(C1CCCCC1)C)NCC#CCC 53587,N1(CC(=O)N(CCNC(C(OC)OC)=O)C2CC2)CC(=O)N1 53588,Cc1nc([N+](=O)[O-])cn1CC(N1CC2C(N(C(=O)COC3CC=CC3)C)C2C1)=O 53589,C1(CCOC)(C(=O)Nc2cncnc2C)CCN(C(=O)C(C(C)C)SC)C1 53590,C(=O)(CS(=O)c1ccc(Cl)cc1)NCC(C1CC1)NC(=O)Cc1cnsc1 53591,Cc1oc(C#N)cc1C(N1CCCC(C(=O)NC2(CC(N)=O)CCC2)C1)=O 53592,c1(-n2c(C)cnn2)ccc(C(=O)NCC2CCCC2NC(=O)CC(C)C)cc1 53593,C(=O)(N=c1[nH]onc1C1(CO)CCC(=O)N1)NC(CCC(=O)OCCCC)=O 53594,C(N=c1[nH]c(=NCCCNC(=N)N)[nH]c2cc[nH]c12)c1cn(C)nc1C(F)F 53595,CC12CNC(C(N3CCCC3)=O)(C1)C2c1ccccc1NC=O.CC(O)C(N)=O 53596,c1(C(N(C2CCN(C(=O)C(C)OCC(C)C)C2)CC)=O)cncc(C(C)C)c1 53597,CC1(CNC(C2(F)CCCC2)=O)CCCN1C(C1CCCCO1)=O 53598,CS(=O)(=O)c1ccc(CSCC(=O)NCc2nc3ccccc3s2)s1 53599,N1(C(CC=CCC)=O)CCN(c2ncncc2C)CC1C 53600,C1(C(=O)N(C)Cc2nnc(O)o2)(NC(C2C(C(C)C)C2)=O)CC1(C)C 53601,C(=O)(C1CCCc2scnc21)NC1CCC(CNC(c2coc(Br)c2)=O)C1 53602,C(=O)(CC(C)C(C)C)N(CC(=O)NCc1c(C)noc1C)CC(C)C 53603,C(=O)(CC(O)CN(C)C)NCC(C)CN(C)C(c1cc(Br)n[nH]1)=O 53604,C1(NC(C2(O)CCCC2)=O)CCC(CCNC(=O)C(C2CCOCC2)F)C1 53605,N1(C(C(C)(C)F)=O)CC(NC(c2cc3n(n2)CCC3)=O)C(C#N)C1 53606,c1(C(=O)NC2CN(C(C(C)(C)c3ccc(Cl)s3)=O)CC2F)ncc(F)cc1F 53607,C1(N(C(Cc2c(C)con2)=O)C)CCCCC1NC(=O)C(C)(C)c1cnc[nH]1 53608,N1(C(CC2(CSC)CC2)=O)CCCCC1CN(C(=O)C(C)=C1CC1)C 53609,N1(C(c2c(C)nc(O)nc2C)=O)CCC2(CC1)CN(C(=O)CC13COC(C1)C3)C2 53610,c1(C(=O)NC2C(NC(C3C(C(C)C)CCO3)=O)C2)ccccc1[N+](=O)[O-] 53611,c1(C(N(C2CCCC(NC(c3ccc(C)s3)=O)C2)C)=O)cc(C)c(C#N)cn1 53612,c1(C(C(=O)NCC(C)CC2CC2)NC(=O)CN(C)C(N)=O)cccnc1 53613,C(=O)(C#CC1CCCCC1)NCC(C1CCCC1)NC(C1C(C)OCCC1)=O 53614,N1(C(C(C)Cc2ccco2)=O)CC(C(N2CCS(=O)CC2)=O)CC(F)(F)C1 53615,N1(C(c2n[nH]c(CC)c2Cl)=O)CC2(CCCC(CNC(c3oncc3C)=O)O2)C1 53616,C1(CNC(C=Cc2cc(OC)ns2)=O)CC2CC(C1)N(C(=O)CC(C)C)C2 53617,C1(CCC)CN(C(=O)C(C)(C)COC(C)C)CCN1C(C1CCCS1)=O 53618,N1(C(CC(C=C)C)=O)CC2(C1)CN(C(c1nnn(CC)c1CC)=O)CC2CO 53619,CC(C)CC(C)(CNC(=O)CN(C)C(=O)C1CC1)NC(c1cnc(O)c(Cl)c1)=O 53620,c1(C(=O)NC(C(=O)OC)Cc2cn(C)cn2)cnn2c(Br)cccc12 53621,C(=O)(C(C)C(O)CCCC)N(CCCCCC(=O)N1C(CCC=C)CCC1)CC 53622,N1(C(CCC(CC)NC(c2cnn3c2OCC3)=O)=O)CCCC2(CCCO2)C1 53623,Cc1cc(C(N2CCOCC2CC(=O)N(C)CC2CCCOC2)=O)cc(O)c1 53624,C1(NC(c2c(C)sc(O)n2)=O)CCN(C(=O)C(C)Cc2ccco2)C(C2CC2)C1 53625,c1(CC(=O)NC(C)CC2CCN(c3ccnc(C#N)n3)CC2)cc(Cl)ccc1Cl 53626,Cn1cncc(C(=O)NC2COCCN(C(c3cnn(C4CCC4)n3)=O)C2)c1=O 53627,N1(C(CCN(CCC)C)=O)CC2CN(C(=O)CC(CC)C3CCC3)CCC12 53628,Cc1cc(C(=O)NCC2CC3CC3N2C(c2ccc[nH]2)=O)c(C)cc1Br 53629,CCCS(=O)(=O)C(C)C(=O)NC1C2CC1N(C(c1cc3cccn3cn1)=O)C2 53630,c1(OC)ccc2c(c1C(=O)NCCN(C(=O)C1=CCCSC1)C1CC1)CCC2 53631,c1(C(=O)NC2C(NC(c3cccc(C(C)(C)C)n3)=O)CCC2)cc(F)ccc1Cl 53632,N1(c2nccc(N3CC=C(C)C3)n2)CCCC2(CC=CCO2)C1 53633,c1(C(=O)NCCN(C(=O)CCn2cccn2)C)ccc2cc(F)c(F)cc2n1 53634,C1(C(=O)NCC2N(C(c3c(OCC)ccs3)=O)CCC2)CCCC2(CCC2)O1 53635,C1(C(N(C2CCN(C(=O)CCN(S(C)(=O)=O)CC)C2)CC)=O)CC2(CSC2)C1 53636,c1(C(=O)NC(CCC2CCC2)C(=O)NC2CC(Cl)(Cl)C2)ccc2nccn2c1 53637,c1(C(=O)NC2C(CC)N(C(=O)Cc3nc(=N)[nH][nH]3)CC2)cnn2c(C)cccc12 53638,c1(C(N)=O)oc(CNCc2nncs2)nc1-c1ccccc1 53639,c1(C(=O)NC2CCC(CNC(c3cnc(Cl)nc3)=O)CC2)ccc(I)cc1Cl 53640,C(=O)(CCCC(F)F)NC(c1ccc(CC)cc1)CNC(=O)Cc1nnc(O)s1 53641,C(CCCCC(=O)O)N(C(C1C(OC)CCC1)=O)C 53642,c1(C(C)C)cccc(NC(C2CC2CNC(c2cccc(SCCO)c2)=O)=O)c1 53643,c1(C(=O)NC2(CC=C)CN(C(C3SCCC3C)=O)C2)ccn2ncc(C)c2n1 53644,C1(CC(=O)NCCNC(=O)NC)CN(C(=O)CC(C)(C)C)CCO1 53645,C1(C(=O)NCC(C)(C2CC2)NC(=O)CSC(F)(F)F)CC1[N+](=O)[O-] 53646,C1(C(=O)NCC(c2ccccn2)C)C2Cc3ccc(Cl)cc3C12 53647,C(=O)(C(F)CC(C)(C)C)NCC(=O)NCC(=O)Nc1ccc(CC)cn1 53648,N1(C(C2C(CC)C2)=O)CCCN(C(c2c(OC)cccc2C)=O)C(C)C1 53649,O(C1(OCC)c2cccnc2CCC1NC(c1csc(O)n1)=O)CC 53650,N1(C(CC2(C)CC2(Cl)Cl)=O)CC2C3CCC(C2C1)N(C(=O)CN1CCCC1=O)C3 53651,N1(C(C=CC=CCC)=O)CC(N=[N+]=[N-])CC1C(=O)NC1CCC(CCO)CC1 53652,Cn1[nH]nnc1=NC1CC2CCC1N(C(C1Cc3nccnc3C1)=O)C2 53653,C1(CNC(=O)C(F)=C2CCC2)CC2CCC1N(C(C1(O)CCSC1)=O)C2 53654,C1(OC)CC(NC(=O)Cn2ccc([N+](=O)[O-])n2)C12CCN(C(=O)C(F)=C(C)C)CC2 53655,c1(CN(CC(=O)NCCCN(C)C)C)ccc([N+](=O)[O-])o1 53656,C1(NC(C=C(C)C)=O)CCOC(CNC(c2ccc(F)cc2)=O)C1 53657,C(CCCC(C)(C)C(=O)NNC(=O)C(C)(C)O)NC(CCC(=O)NS(C)(=O)=O)=O 53658,Cc1cc(C#N)ccc1C(N1CCC(N(C(=O)CNC=O)C)C(C)C1)=O 53659,N1(C(c2cncc(C)n2)=O)CCCC(CO)(NC(c2cc(C(F)F)ncn2)=O)C1 53660,Nc1c(C(N2CC(CNC(c3ccon3)=O)C3CC23)=O)cnn1-c1ccccc1 53661,C(C(O)C(=O)NC(C1CCCN1C(c1cc(C(C)C)on1)=O)(C)C)SC 53662,N1(C(C2(OC)CC2)=O)CCC(C2CC2NC(=O)CN(CC(C)(C)C)C)CC1 53663,N1(C(Cc2c(SC)cccc2)=O)CC(C)CN(C(=O)C=C(C)C)C(C)C1 53664,C1(CCNC(c2ncn(C(C)C)c2)=O)CN(C(=O)C(c2cncnc2)C)CC1C 53665,c1(C(c2nnnn2C)NCC(CCC)C)cc(S(N)(=O)=O)ccc1F 53666,c1(C(N(C(C)CC2CC2)C)=O)cc(CNC(C2(C3CC3)CCC2)=O)ccn1 53667,C1(CC(=O)NC2(c3cccs3)C(C)C2)CCCS1(=O)=O 53668,N1(C(c2n(CCC)ccc2)=O)CC(C(=O)NC2(C(=O)NC)CC2)CC(C)C1 53669,C1(NC(C(=O)NCCC(OC)OC)=O)CCCN(CCN(C)C)C1 53670,C(=O)(C1=CCCOCC1)N1CC(O)(CN(C(C=CC(=O)OCCCC)=O)CC)C1 53671,C1(C)(COC)CC(NC(=O)CCCc2ccccc2)CN1C(=O)CC(C)(F)F 53672,C(C(C)(CN=C(NC(C)C)N1CCCC(N2CCCS2(=O)=O)C1)OC)OC 53673,S(=O)(=O)(CC(=O)NC1(C(=O)NCC2CCCO2)CCSC1)NC 53674,c1(CNC(C(C)C2CCOC2)=O)cnn2c1CN(C(=O)CC13CC(C1)C3)CC2 53675,N1(C(C2C(OCC)C2C)=O)CC2(CCN(C(C3CC4(C)CC3CO4)=O)C2)C1 53676,CCCCC(C(=O)NCCC1(C(C)(C)O)CC1)N(C)C.C12(CC1)C(=O)NC2 53677,Cc1cc(C(=O)NC2CC(NC(=O)C(C)Sc3ccc(Cl)cc3)C2)c(C)s1 53678,C(=O)(C(F)C(=O)NC(CO)C(=O)NC1C(OC)CC1O)OCC 53679,c1(C(=O)NC(CC)CNC(c2c[nH]c(=N)o2)=O)sc2cccc(F)c2c1Cl 53680,c1(NC(N2CCN(c3cncs3)CC2)=O)nc2ccccc2[nH]1 53681,N1(C(CC2(C)CC2)=O)CCC2(CNC(c3ccccc3C3CC3)=O)CCCCC12 53682,Cc1ccc2ccnc(NCc3nc(C(=O)O)c(C)s3)c2c1 53683,N1(C(C=CCN)=O)CCCC(F)(CO)C1.CC(C)(O)CC=O 53684,c1(CC(N2CCCC(NC(=O)Cn3cccn3)CC2)=O)ccc2c[nH]nc2c1 53685,N1(C(C(CC)OC)=O)CCC(C(=O)OC)C1NC(=O)C(F)(F)F 53686,C(=O)(C(O)C1=CCCCC1)NCC1(O)CN(C(C(CCCCC)O)=O)C1 53687,C1(C(N2CC(C)(NC(CCC(=O)NC)=O)C2)=O)CCC(=O)C(C)C1(C)C 53688,c1(C(N(CC(C)N(C(C(C)n2ccnc2)=O)C)C)=O)cc(S(N)(=O)=O)sc1Cl 53689,C12(CNC(C(C)=CC3CC3)=O)CCCC(CN1C(=O)C(O)C(F)(F)F)C2 53690,C12CCCCCN1C(=O)C(C)N(C1CC1)C2=O.C1(CC)CCCC(C#N)C1 53691,N1(C(C(CC)OC2CCCCC2)=O)CCCC2(CCCN2C(C)=O)C1 53692,C1(NC(c2ccc(F)cc2O)=O)C2COCC1CC(NC(C1CCCCS1)=O)C2 53693,c1(C(=O)NCC(CNC(=O)CNS(=O)(=O)C2CC2)OC)cccc(C)c1C#N 53694,C1(NC(CC2(C=C)CCC2)=O)(CO)CCN(C(C2CN(CC)CCO2)=O)CC1 53695,N1(C(C(CC2CCCC2)OC)=O)C2CCC1CC(CNC(C1(CO)CCC1)=O)C2 53696,C1(CCNC(C2(C)CC(=C)C2)=O)CCCN(C(c2cc(CCC)[nH]n2)=O)C1 53697,N(C(=NCCN(C)C)NCc1ncccc1N(C)C)CC(C)(C)OCC 53698,N1(C(c2cc(C)n(C)n2)=O)CCCN(CCNC(C2CC2CF)=O)CC1 53699,CC1(CCCC(=O)NCC2(O)CCN(C(=O)Cc3cccs3)C2)NC(=O)NC1=O 53700,c1(-n2cc(CN3CC(CCC)C(CO)C3)nn2)cccc([N+](=O)[O-])c1 53701,C12(C(N3CC(N(C(CCc4ccc(CC)cc4)=O)C)C3)=O)CC(C)(C1)OC2(C)C 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53754,C(CC(N)CC(=O)NCC1(c2ccccc2)CCCCC1)SC 53755,C1(NC(C2CCCC23CC3)=O)CCCN(C(=O)Cc2cscc2Br)CC1 53756,C(CCC(=O)NC1CCC(CNC(=O)C(F)=CC2CC2)C1)OCC 53757,c1(CC)ccc(C(=O)N(CCNC(c2ccc(C)o2)=O)CC2CC2)c(F)c1 53758,C1(CC(=O)OC(C)(C)C)CCCN(C2=NCCC(OCc3cccs3)N2)C1 53759,CCC1=NOC(C(=O)NCCCCC(C)NC(c2cc(C(C)C)no2)=O)C1 53760,CCCN=C(NCC(CC)C(C)C)NCCOc1nnnn1-c1ccc(F)cc1 53761,CC1CCN(C(=O)CC2CSCCO2)CCN1C(=O)CC1C=NN(C)C1=O 53762,C(C(=O)NNC(=O)CCSC1CCCCC1)c1c(C)n[nH]c1C 53763,C1(CNC(CC2(C)CCN2C(=O)CC2CCCNC2=O)=O)CCC(F)(F)C1 53764,N1(C(c2nccc(SC)n2)=O)CCN(C(C2CCC(C)=C(C)C2)=O)CC(C)(F)C1 53765,c1(C(=O)NCCC(CNC(C2C(=C)C2)=O)O)ccc(OC)c(S(=O)(=O)N)c1.C1N=N1 53766,CCC(CC)C(F)C(=O)N1CC(C(=O)NC(C2CCC2)C2CC2)C2(CCC2)C1 53767,c1(C(=O)NCCC2CCN(C(c3ccc(CC)o3)=O)C2)cncc2ncn(C)c12 53768,C1(NC(CSC(C)C)=O)CC(NC(C2CC(S(C)(=O)=O)C2)=O)C12CCOCC2 53769,C1(NC(=O)CN2CCCNC2=O)(CO)CCCN(C(=O)CC(C2CC2)C2CC2)C1 53770,C1(CC(=O)N(CCC=C)C(c2ccccc2)=O)C2C=CC3(CN(C(C)C)C(=O)C13)O2 53771,c1(C(N2C(CN(C(C3(OC)CS(=O)(=O)C3)=O)C)COCC2)=O)ccc(O)nc1Cl 53772,C(c1cnn(C)c1)=CC(=O)NC1(CO)CN(C(c2c(OC)csc2)=O)C1 53773,c1(CNC(C(C)Cc2ccccc2)=O)ccc(-c2cc(CO)ccn2)cc1 53774,C1(NC(c2cn(CC=C)nc2)=O)CN(C(C2CCCCC2(F)F)=O)CCC1CO 53775,O=C1COC(CNC(C2CCN(C(=O)C(F)C3CCC3)CC2)=O)CN1 53776,c1(C(=O)NCC2(NC(C(CC#C)C)=O)CCOC2)cc(C(N)=O)ccc1F 53777,c1(C(=O)NCC2(F)CN(C(c3c(CC)nc[nH]3)=O)C2)ccc(C2(C#N)CC2)cc1 53778,N1(C(c2ccn(C(CC)CC)n2)=O)CC(CNC(c2cc(OC)no2)=O)C2CC12 53779,c1(CNCc2ccc(-c3ccc(OC)cc3)o2)n[nH]c2ccc(C)cc12 53780,C(=O)(CCCCNC(=O)C1CC1)NC(CNC(C(C)(C1CC1)OC)=O)C(C)C 53781,C(c1ncco1)=CC(=O)NCC1CCN(C(c2ccoc2C2CC2)=O)C1 53782,CC(C)(C)C1=NOC(C(=O)NCCOCCNC(=O)C(F)CC2CCOC2)C1 53783,C1(OC)CN(C(=O)C(C#N)C2CC2)CC1NC(=O)CCC1CCCC1 53784,Cn1cc(C(N2CCC(CO)C(NC(=O)CC3CC4CC4C3)C2)=O)c2sccc12 53785,C1(NC(c2c(C)cc(C)o2)=O)(CO)CCN(C(C2CC(=O)C2(C)C)=O)CC1 53786,C1(C(=O)NCC2=CCCCC2)C2CCN(C(c3ccsc3Cl)=O)CC12 53787,C1(CC)(NC(c2coc(C(C)(C)C)n2)=O)CCCN(C(C2CSCCS2)=O)C1 53788,c1(C(C)=O)ccc(C(=O)NC(CNC(=O)CCC(F)F)CC(F)(F)F)cc1F 53789,C1(C(=O)NCC(C2CCCC2)NC(C(CN(CC)CC)F)=O)CCC(C)CC1 53790,N1(C(c2cnn(C(CC)CC)c2C)=O)CCC(C)C(NC(c2csc(=N)[nH]2)=O)C1 53791,NS(=O)(=O)CCC(=O)NCCNC(C1CCCN(C(c2cnns2)=O)C1)=O 53792,c1(C(N2CC(O)(CNC(CC3C(C)C3)=O)C2)=O)cc2c([nH]1)CCCC2=O 53793,C=C=C(C)CC(=O)N(C1C2CCN(C(=O)CCC(=O)C3CC3)C12)C1CCN(C)CC1 53794,C#Cc1ccccc1CNC(C1CCN(C(=O)C(C)C=CCC)CC1O)=O 53795,c1(C(=O)NCc2c(C(N(CC(CC)OC)C)=O)cco2)cncnc1C 53796,N1(C(Cc2c(C)ccnc2)=O)CCCC(C(=O)NC(c2nc(=O)o[nH]2)C)CC1 53797,c1(CC)ccncc1CNC(c1cccn1C)c1nnnn1-c1ccccc1 53798,N1(C(C(C)N(CC)CC)=O)CCN(C(c2cc(C(C)=O)cn2C)=O)CC(O)C1 53799,Cc1nccc(C(=O)NCC2(F)CC(CNC(=O)C=CC3CCCO3)C2)n1 53800,N1(C(CN(C(=O)CCC(F)(F)F)CC)=O)CCCC(C)(N(C)C)C1 53801,C1(CS(N2CCN(c3nccc(OC(C)C)n3)CC2)(=O)=O)CC2(CCNCC2)C1 53802,N1(C(Cn2nc(C)c(Cl)c2C)=O)CC2(CCCCN2C(c2nn(C)cc2Cl)=O)C1 53803,C(CC(C(N)=O)NC(C1(NC(C2CC2(Cl)Cl)=O)CCOCC1)=O)OC 53804,N1(C(CC2CC(C)C2)=O)C2CCC1CN(C(C1CCn3nncc3C1)=O)C2 53805,c1(N2CC(C(C)NC(c3ccc(CO)o3)=O)OCC2)ncccc1C#N 53806,c1(C(=O)NCCCCCN(C)C(C2C=CCC2)=O)cnn2c1OCC(O)C2 53807,CCCCCC(F)C(=O)N(C(C)C(=O)NOCCCO)C 53808,Cc1nsc2ncc(C(=O)NCC3(F)CCN(C(=O)CCCC(C)(C)C)C3)cc12 53809,c1(C(N2CC(NC(c3cc(OC)n[nH]3)=O)C(C)(C)C2)=O)nn(C)cc1S(C)(=O)=O 53810,C12(C(N3C(CNC(c4ccccn4)=O)C4CC4C3)=O)CCC(F)(CC1)CC2 53811,Cc1ccc(F)c(C(=O)NCC2CC(F)(CNC(c3ccn(C)c3C)=O)C2)c1 53812,c1(C(=O)NCC2CCC(NC(C(C)OC3CCCC3)=O)C2)cc(Cl)c(Cl)cc1N 53813,C(=O)(C(C)(C)C(F)(F)F)NC1CCCN(C(C(C2CCCC2)NC(C)=O)=O)CC1 53814,C1(C2CC2)(NC(CC(C)N(C)C)=O)CCN(C(c2coc3c2CCCC3)=O)C1 53815,CN1CCN(C(=O)Cc2cnns2)C(CNC(=O)CC2CCCCC2(C)C)C1 53816,c1(COC2C(OC(C)=O)C2)nc2sc3c(C(C)(C)OC)c2c(=O)n1CCCC3 53817,C12(CNC(CCCOCC=C)=O)CC1CN(C(=O)C(C)Cc1cnc[nH]1)C2 53818,C(N=c1nc2scnc2c(N2CCCC(CC(F)F)C2)[nH]1)C1OCC(C)(C)OC1 53819,CC1(C)CCC(CNC(C2CCC(=O)NC2)=O)N(c2nnco2)C1 53820,c1(C(N(C(CNC(C2(C)CCC(C)C2)=O)C2CC2)C)=O)occ2c1CCOC2 53821,CS(=O)(=O)CCCC(=O)N1CCC(O)(CNC(=O)C=Cc2cscn2)C1 53822,N1(C(=O)Nc2n(C)ncc2C2CCC2)CC2C3CCC(C(O)C3)C2C1 53823,C(CCC(C)C(=O)N(CCCN(C(=O)Cn1cnc([N+](=O)[O-])n1)C)C)OC 53824,c1(C(=O)NC)ccccc1OCc1cscc1Br 53825,C1(NC(C(COC)C)=O)CN(C(=O)CC2CCCC2)C(C)(C)C1 53826,C1(C(=O)OC)CC(C(=O)NCCCCNC(=O)C(C)(C)C2CC2)C1(C)C 53827,c1(OC)cc(F)cc(C(N2CCOCC(CNC(=O)C3=NOCC3)C2)=O)c1N 53828,c1(C(=O)NC23CCN(C(=O)CCC4CCOCC4)CC2C3)c[nH]c2nccc-2c1 53829,c1(C(N(CCCC(=O)N(CC(=C)C)CC(=O)N(C)C)C)=O)ccc(C)c(F)c1 53830,S(=O)(=O)(c1cc2sc(=NCC3=CCCC3)[nH]c2cc1Cl)NC(c1ccc(Br)c(C)c1C)=O 53831,c1(C(C)OC)nc(C)c(C(N2CC(CNC(=O)C=CSC)C(O)C2)=O)s1 53832,CC(C(=O)N(C1CN(C(=O)CC(O)CCC)CCC1O)C)S(N)(=O)=O 53833,C1(CN(C(c2n(C(C)C)ncc2)=O)C)CN(C(=O)CC2CN(C)C2)CCO1 53834,C(=O)(C#CC1CCCO1)N(C)CC1(O)CCN(C(c2nn(CC)c(O)c2)=O)C1 53835,Cc1ccc(-c2csc(NC(CNC(C3(N(C)C)CC3)=O)CO)n2)cc1 53836,C(=O)(C(C)CC(C)C(C)=O)NC(CNC(c1c(CC)n(C)nc1)=O)CCOC 53837,C=CCCCCCC(=O)N(C1CCCCN(C(=O)C(C)(C)OCCC)C1)C 53838,N1(C(C2(C)CCCC2O)=O)CC2(CC(CNC(c3cccn3C3CC3)=O)C2)C1 53839,C1(NC(C=CCCC)=O)CC1C1CCCN(C(=O)Cc2ccccc2OC)C1 53840,C1(NC(C(C)=CC2CC2)=O)C(C)CN(C(=O)CC2(C)CCCCC2)CC1C 53841,c1(C(=O)OCC)c[nH]c(=NC2CCC3CCC23)cn1 53842,C1(NC(C(CSCC)NC(c2[nH]nnc2C)=O)=O)CCCCC1F 53843,Cc1cc(N)cc(C(=O)NCC(C)N(C(=O)CCc2cnn(C)n2)C)c1F 53844,N1(C(c2c(C)nc(C)o2)=O)CCCC(C(N2CCC(CC(F)F)C2)=O)C1C 53845,C(=O)(CC1=NN(C)C(=O)C1)NCC(CN(C)C(C1CCCSC1)=O)(C)C 53846,C=CCCCC(C)NC(C1C=CCCN1C(c1cc(C)oc1C)=O)=O 53847,c1(NC(C2N(Cc3ccc(C)nc3)CC2)=O)cccc([N+](=O)[O-])c1F 53848,NC(=O)CCC(=O)N1CC=CC1CNC(c1csc(Br)c1Cl)=O 53849,Cc1ncc2ccc(C(=O)NC3CC(NC(c4cccnc4)=O)C34CCC4)cn12 53850,C1(C(N(CC(=O)NC(C#C)CC2CC2)C)=O)CCCOC1 53851,C1(C(N(C(C)C)C)=O)CCN(C(c2ccc(OCCO)cc2)=O)C1C.C1C(=O)O1 53852,c1(C(=O)NC2CCC(CNC(C3ON=C(C)C3)=O)C2)ccc2c(c1)CC(C)O2 53853,N1(C(C(=O)NCCSC)c2cccs2)CCc2c(Cl)cc(Cl)cc2C1 53854,Cn1cc(CNC(=O)C(=O)NC2CC3CCC2O3)c(-c2ccnn2C)n1 53855,C1(CNC(=O)CC2C=CCCC2)(NC(C2CCCCC2O)=O)CCCCC1 53856,c1(C(N2CCC(CC(C)NC(C3CC(F)C3)=O)CC2)=O)ccc(Cl)c(C#N)c1 53857,Cc1cc(C(=O)NC2CCOCC2C(=O)N(CCCO)C2CC2)c(C)n1C 53858,Cc1nc(CC2CC2)sc1C(=O)NCCC1CCC(NC(c2c[nH]nc2F)=O)C1 53859,C1(NC(c2ccccc2F)=O)CN(C(c2ccc(C3CCOC3)s2)=O)CC1F 53860,C1(C(=O)NC(CN(C(=O)CS(N)(=O)=O)C)(CO)CO)CC12CCOCC2 53861,C(=O)(C1=CSCCO1)NC1C(CNC(=O)Cc2cc[nH]n2)CC1 53862,c1(C(N(C2CC(NC(C3CC3c3ccn(C)n3)=O)C2)C)=O)nccnc1N 53863,CC1CC(N(C(=O)C(F)C2CC(NC(c3c[nH][nH]c3=N)=O)C2)C)CCO1 53864,c1(C(=O)NC2CC(CNC(C(C)OC)=O)C(O)C2)ncc(Cl)cc1F 53865,C12(C(N3C(C4CCN(C(c5ccn(C)n5)=O)CC4)CCC3)=O)CCCC1C2(F)F 53866,C(=O)(C1=NOC2(CCC2)C1)NC(CCC)CCCNC(=O)C(C)(F)F 53867,CC1CCC1C(=O)NCCCNC(N)=O.C12CC(C1)OCC(=O)N2 53868,C(=O)(CC(C(F)F)NC(c1cnco1)=O)NC(C)(C)C(F)F 53869,c1(C(N2C3CC(NC(=O)CCOC4CC4)CC2CC3)=O)ccc(F)c2[nH]ccc12 53870,C1(C(=O)NCCN(C(=O)CCNCCCNC(N)=O)C(C)C)(OC)CCC(C)C1 53871,N1(C(c2c(CC)con2)=O)CC2(CCN2C(=O)CCN2CCC(F)C2)C1 53872,c1(SCC(=O)NCCOCCCN(C)C(c2ccccc2)=O)ccccc1F 53873,c1(CCC)onc(C)c1C(=O)NCC1(C)CCC(NC(c2ccc(C)cn2)=O)C1 53874,N1(C(c2n(C)nc(O)c2)=O)CCC2(CC1)CC2C(N1CC2CCC(CC2)C1)=O 53875,N1(C(CN(CC)CC)=O)CCCC12CCN(C(=O)C(C)CC1CC1)C2 53876,C1(C(N(C2CCOC2=O)C)=O)CN(C(c2ccn(CCF)n2)=O)CC1(F)F 53877,C1(O)(CN(C)C)CCN(C(C2(NC(C3CC3(C)C)=O)CC2(C)C)=O)C1 53878,C1(n2cc(CNC)nn2)CCN(C(C23CCCC2CC3)=O)CC1 53879,C(=O)(C1=NN(c2ccccc2)C(C(N)=O)C1)NCC1N(C(CC=C)=O)CCCCC1 53880,CC(CC(C)(C)C)C(=O)N1CCC1CNC(c1ccncc1Br)=O 53881,Cc1ccnc(C(N2CCOCCC2C(=O)NCC2OC(=O)NC2(C)C)=O)c1N 53882,N1(C(CC2C(C)C2)=O)CCC2(CC1)CCN(C(C1CC13CC(C)(C)C3)=O)CC2 53883,c1(C(=O)NC2C(CNC(CC3(C(=O)OC)CCC3)=O)C2)cc(F)ccc1OC 53884,c1(C(N2CC3CC(NC(Cn4c(C(C)C)ncc4)=O)C3C2)=O)ccn2nccc2n1 53885,C(CCOC)(C(=O)NC1(CSC)CCC1)NC(C(C)OCC=C)=O 53886,C(=O)(C(CCC(C)C)NC(=O)C1=CCC(C)CC1)N(C)Cc1nc(C)[nH]n1 53887,CC(C)C(CCN(C)C(C)=O)NC(c1ccc(-c2ccccn2)nc1)=O 53888,Cc1cc(C(=O)NC2CC3C(NC(=O)Cc4sccc4Cl)C3C2)c(C)n1C 53889,c1(CC(C(=O)N(CCCNC(C2(CC#C)CCCO2)=O)CC)C)ccc(F)cc1 53890,Cc1ccc(S(=O)(=O)NC2CCC(C(=O)Nc3ccccc3CO)CC2)cc1Cl 53891,C1(CNC(C(C)Cc2ccncc2)=O)CC2(CC2)CN1C(c1nccnc1N)=O 53892,CCC(CC)CC(=O)NC1CCN(C(c2cccc(N)c2O)=O)CC1F 53893,c1(C(=O)NC2CC3CN(C(CSCCCC)=O)C(C2)C3)cccc2nc(O)[nH]c12 53894,C(N=c1[nH]c2c(c(=NC3CCSC3)[nH]1)CCC2)c1ccc(N)cc1 53895,C1(NC(C=CC(C)(C)SC)=O)CN(C(=O)CCc2ncc[nH]2)CC1C(F)F 53896,C1(CN(C(=O)C=CC2CCCO2)C)CCN(C(c2cnoc2-c2cccs2)=O)C1 53897,Cc1ccc(CNC(=O)CC2CC(C)N(C(=O)C(C)CC3CC3)C2)c(C)c1 53898,Cc1ccc(CCNC(=O)C(C)CNC(=O)C(n2ccnc2C)C)cc1 53899,c1(C(N(CC(CC)NC(=O)COC2CCCOC2)C)=O)ncc(C)cn1 53900,c1(CN(C(=O)CN2CCSCC2)CCNC(C2CC(C#N)C2)=O)cccc(Cl)c1 53901,N1(C(CC(C)C2CCCCC2)=O)CCC(NC(=O)CSC2CCOC2=O)C(C)(C)C1 53902,c1(C(N(CC(C)N(C(=O)Cc2cccc(F)c2F)C)C)=O)cc(F)ccc1F 53903,c1(C(=O)NCC(C(C)C)(C)NC(C2CC=CCO2)=O)cc2cn[nH]c2cn1 53904,c1(NC(C2CCC(CNC(C(C)O)=O)CC2)=O)ccc(S(N)(=O)=O)cc1Cl 53905,CC1(C)OC2(CC(c3ccc(F)c(O)c3)=O)CCC1(C(=O)O)CC2 53906,CC(O)C(C(=O)N1CCC(C)(NC(c2cnn(-c3cccnc3)c2)=O)C1)N(C)C 53907,c1(NC(C(CC2CC2)NC(C(CC2CCC2)OC)=O)=O)cnc(C)c(Cl)c1 53908,c1(CCC(=O)NC2CN(C(=O)CC34CCCC3C4)CC2O)cccnc1F 53909,C(CN=c1[nH]c2cccc(F)c2s1)(C1CC1)NC(=O)C#CC1CCCCC1 53910,CS(=O)(=O)c1ccccc1C(N1CCCCC(NC(=O)C2=COCCC2)C1)=O 53911,C1(NC(CC(C(C)OC)NC(=O)Cn2ccccc2=O)=O)CC2(CNC(=O)O2)C1 53912,C1(CC)CCCCC1OCC(=O)NCC1CCC1NC(c1nc(C(C)C)cs1)=O 53913,C1(OC)CN(C(=O)CC2CCC=CCC2)C(C)(CNC(=O)Cc2csnc2C)C1 53914,CN1C(=O)OCC12CN(C(=O)NCc1ccnc(OC3CCCC3)c1)C2 53915,CC(C)C(C)(O)C(=O)N1CC(CNC(C2CCC3CCC2O3)=O)C1 53916,N1(C(CCC(C)SC)=O)CC2CCCC2(NC(=O)Cc2ccn(C)n2)C1 53917,N1(C(C(C)Cn2cncn2)=O)CCCC(C(N2CC(CC34CC(C3)C4)C2)=O)C1 53918,c1(C(N2CC3(C(=O)O)CCC2CC3)=O)cc(=O)c2ccccc2[nH]1 53919,N1(C(c2cc(C(CC)CC)no2)=O)CCC2CCN(C(C3CCOC3C)=O)CC12 53920,c1(C(N(C2CCN(c3ncc(Cl)c(O)n3)CC2)CCC)=O)coc2c1COC2 53921,C(=O)(CCCC(=O)N(CCCN(C(=O)CN1CC(C)C1)C)C)NCCC 53922,N1(C(c2cccc(NC)c2)=O)CCC(C2CC2)(CNC(C2CN(C(C)=O)C2)=O)C1 53923,CC(C)CCC(=O)NCC(=O)NC1CC(CNC(c2ncn(C)n2)=O)C1 53924,C(=O)(C(O)CCNC(=O)C=CC1CCOC1)NCCOCCOC 53925,N1(C(=O)CNC(C2(n3nccn3)CC2)=O)CCC(C2CCCC2)C1 53926,C(=O)(C(C)CCN(C)C)N1CC2(C1)NC(=O)CC(=O)NC2.C#CCOC 53927,c1(CSC)ccc(C(=O)NC(C(=O)NCC2CC2[N+](=O)[O-])C2CCOC2)o1 53928,N1(C(c2cncc(CC)c2)=O)CC(C)CCC1CNC(=O)CCc1nc(O)n[nH]1 53929,C#CC1(C(N2CC(CC(F)F)C2)=O)CCN(C(=O)C(C)C2CC2)CC1 53930,c1(COC)nc(C(=O)NC(C)C(CO)NC(=O)C(F)=C(C)C2CC2)n[nH]1 53931,C1(C(=O)NCC(F)(F)C(C)(C)O)(CC)CCCN(C(=O)C=Cc2ccco2)C1 53932,N1(C(CC=C=C)=O)CCC(C(=O)NC2C=CCCC2)C1(C)C 53933,CCN(CC1CC1)N(C)CCCN(c1ccccc1)C(C1CCCCC1)=O 53934,Cc1c(C(=O)N(C2CCCCN(C(C3CCCS3(=O)=O)=O)C2)C)cccc1F 53935,c1(C(=O)NCC2(CCNC(CC3C(C)CCC3)=O)CC2)c(F)cc(F)cc1Cl 53936,C1(CC)(CC)CC(O)CN1C(=O)C(C1CCN(C(c2cc(F)n(C)n2)=O)C1)F 53937,n1(CCCOC)nnnc1C(COC1CCCCC1)NCc1cc[nH]n1 53938,C1(CNC(C2(CC)CC2(F)F)=O)CN(C(=O)CCc2cccn2C)CCC1(C)C 53939,C1(N(C(C(CC#C)C2CC2)=O)C)CN(C(c2ccc(C(N)=O)cc2)=O)CC12CC2 53940,C1(NC(C(C)=CC)=O)CCN(C(=O)Cc2nonc2C)CC1O 53941,C1(CNC(C2CN(C)C2)=O)CC(NC(c2ccc(Cn3cccn3)o2)=O)C(O)C1 53942,C1(C)(NC(C(N2CCCC(C)C2)=O)=O)CCCN(C(c2ccnc(O)c2)=O)C1 53943,Cc1nc2cccc(C(=O)NCC3CC3NC(C3(CC(C)C)CCCC3)=O)c2[nH]1 53944,CC1CCOC1C(=O)N(CCCO)Cc1cn(C2CC(N(C)C)C2)nn1 53945,N1(C(C(C)CC2CCCC2)=O)CCCCCC1CNC(=O)CCCCCN(C)C 53946,N1(C(c2ccc(NC)cc2)=O)CCCCC(CNC(=O)C(C)CN2CCCC2)C1 53947,c1(CC)nccnc1C(=O)NCC(C)CC(=O)N(C1CC2CCC1O2)C 53948,C(=O)(C1=CC2CCCCCC12)N1CCC(C(C)NC(c2ccc(C(C)=O)s2)=O)C1 53949,C(c1ccc(S(=O)(=O)NC)cc1)=CC(=O)NCC(CC=C)NC(=O)CC1CC1 53950,C=CCCC(C(=O)OC)NC(=O)C(C)SC.C12(CCSC1)C(=O)N2 53951,C1(C(=O)NCCCNC(c2ccc(OC)nn2)=O)CCN2CCCC2C1 53952,Cc1nsc(C(N2CC(F)(CNC(=O)CSC(F)(F)F)C2)=O)c1N 53953,O(C1CCc2c(Br)cccc21)C(=O)C(c1ccc(F)c(F)c1)=O 53954,N1(C(C2(F)CCN(C(C(C=CC)O)=O)C2)=O)CC(C)OC(C)(C)C1C 53955,C1(C)(C(=O)NCCN2CCN(C(C3OCCC(C)C3)=O)CC2)CCS(=O)(=O)CC1 53956,c1(C(N2CC(c3ccc(C)cc3C)OCC2)=O)cc(N)cc(O)c1Br 53957,c1(C(=O)NCCC2(CNC(C3CC3C(=O)O)=O)CC2)cc2c(cn1)CCCC2 53958,Cc1nsc(Br)c1C(=O)N(C)CC1CCCCN1C(=O)CCC1(C)CC1 53959,N1(CC)CCN(C2CN(C(C)COC)C2)CC1.C(C)(C(=O)NCC)OCCO 53960,Cc1c(NC(c2ccnc(O)c2)c2nnnn2CC(F)F)ccc(Br)c1Cl 53961,C1(CNC(CCCCC#C)=O)CCCC2CN(C(=O)Cc3ccc(F)nc3)CC12 53962,n1(CC(=O)N(C2CN(C(=O)COCCN(C)C)CC2F)C)cnc2ccccc12 53963,Cc1cnn(CC(=O)NC2CC(CCNC(=O)C(C)Oc3cccnc3)C2)c1 53964,CCC(CC(=O)NCC1OCCC1C(=O)NCc1cc(OC)no1)C(F)F 53965,N1(C(C2C(C=C)OCC2)=O)C2CCC1CC(NC(=O)C(C)(C)c1cncnc1)C2 53966,N1(C(C2C(C)=C2)=O)CC2CCCC(C1)N2C(=O)CC(C)c1ccco1 53967,C1(C(=O)NC(CCNC(Cc2ccn(C)c2)=O)(C)C)CCNC(=O)C1 53968,C(=O)(C1=Cc2ccccc2C1)N(CCC(=O)NC1COCCC1O)CC=C 53969,C(=O)(C1=C(Cl)CC1)NCC1CC1COC(N(CC(O)C(=O)OC(C)(C)C)C)=O 53970,N1(C(CN(CCC)C)=O)CCC2(NC(C3CCN(C(C)=O)CC3)=O)CCCCC12 53971,C=C(C)C1CC(Nc2cc(F)cc(Br)c2F)C(C)C(C#N)C1 53972,N1(CC(=O)CCC2CC2(F)F)CCC(NC(=O)C(c2ccc(Br)cc2)(F)F)CC1 53973,c1(C(=O)NC2(C)CCC(NC(=O)C#CC3CC3)CC2)cc[nH]c(=N)c1[N+](=O)[O-] 53974,Cc1ccc(CC(=O)NCC2CCN(CCN(C3CCCO3)C3CC3)C2)c(C)c1 53975,N1(C(c2c(CC)nc[nH]2)=O)CC2CCC(C1)C2CNC(=O)C(C)NC(=O)COC 53976,C12(C(NOCC(C(C)C)O)=O)CCC(NC(=O)Cc3cncnc3)(CC1)C2 53977,CC(C)CC(CNC(=O)C1=CCCOCC1)C(=O)N1CCc2n[nH]cc2C1 53978,C(=O)(CC(O)CNC(C1CCCC1O)=O)NCC(=O)N(CC)CC 53979,Cn1nc(C(N2CCC(C)(NC(C3CCCC3)=O)CC2)=O)c2cc(F)ccc12 53980,c1(CC)ccc(C(C)C(=O)N(CCNC(=O)CC(C)C2CCCO2)C(C)C)cc1 53981,C(=O)(C(CC(C)C)N(C)C)NCC1(OC)CCN(C(c2ccn(C3CC3)n2)=O)C1 53982,C(=O)(C1=CCCC1(C)C)N1CC2C(NC(c3cn(C)nn3)=O)(CC2)C1 53983,c1(C(N(CCCNC(=O)Cc2ccnn2C)CC)=O)cnc(Cl)c(F)c1N 53984,c1(COCC)nnc(N2CCCC2CCNC(=O)C2CC2)s1 53985,CC1CC(NC(c2cc(C#N)n(C)n2)=O)CCN1C(=O)Cc1cnc(C2CC2)[nH]1 53986,C=CCN(OC)C(=O)CCC1CCCN(C(=O)CC2CC(F)(F)C2)C1 53987,C(C1=NOC2(CCC2)C1)NC(C1CCN(C(C(CC)N(C)C)=O)C1)=O 53988,Cn1ccc(-c2cc(C(=O)NCC3CCN3C(=O)CC3CCCO3)n[nH]2)c1 53989,c1(OC)cc(CC(=O)NCCc2ccc(-c3ccccc3)[nH]2)cc(OC)c1O 53990,C1(C(=O)NC(c2nccn2C)CC)CCCN(C(c2nn(C)cc2C)=O)C1 53991,C1(N(C)C)(C(=O)NC2CCCC(N(C(=O)C=Cc3cc[nH]n3)C)C2)CCCCC1 53992,c1(C(=O)NCCN(CCC)C(C2(C)CC(C)=NO2)=O)nc(C)n(C)n1 53993,Cc1nc(CC(=O)NC(Cc2cn[nH]c2)C(=O)NC2(C)CC2)n[nH]1 53994,C1(NC(CCc2nc(C)c(C)[nH]2)=O)CN(C(=O)CC2CCCCC2)CCC1C 53995,c1(-c2cc(NC(C3CCCCCC3)C)sc2)ccc(F)cc1 53996,c1(C(=O)NC(C)CNC(C2CCN2S(C)(=O)=O)=O)cnc2n1CCS2 53997,C1(CNC(CCCOCC=C)=O)C(C2CC2)CCN1c1nccn2nnnc12 53998,CCCCC(CC)CC(=O)NCCCCCCN(C(=O)C(CC)C(C)(C)CC)C 53999,c1(CC(C(=O)N(CCOCCNC(C2(CC)CCOC2)=O)C)C)ccccc1Cl 54000,C1(C(=O)NCC2N(C(c3cc(C)sc3C)=O)CC(F)C2)CCCC2(CC2)C1 54001,C1(CNC(C(c2c(F)cccc2F)(C)C)=O)C2CCC(C2)C1N 54002,C1(NC(c2c(COC)cc[nH]2)=O)CC(C)CN(C(=O)COCCF)C1 54003,Cc1cc(Br)ncc1NC(C1CC(O)CN1c1ccncn1)=O 54004,N1(C(C2CN(C(Cc3cccc(C)n3)=O)CC(F)C2)=O)CCC(O)C(C)(CO)C1 54005,c1(NC(C)C)ncccc1C(=O)NC1CCCC1NC(C1CCOC1C1CC1)=O 54006,c1(C(=O)NCCN(CCOC)C(C2OCCC2C)=O)cc(C)ncc1Br 54007,Cc1cc(F)ccc1C(=O)NC1C=CCCC1C(=O)NCC(F)Br 54008,C(C)(C)(CC(F)C(=O)N(C1CCOC(C)(C)C1)C)NC(C1C(C)OC(=O)N1)=O 54009,CC1(C)CC=C(C(=O)NCC(C)(C2CC2)NC(c2ccc(O)nn2)=O)CC1 54010,C1(CNC(c2c(C(C)C)nns2)=O)CCN(C(C2CN(C)CCO2)=O)C12CC2 54011,C1(N(C(CCN(C(=O)C(C)Cn2cccn2)CC)=O)C)CC1C1CC1 54012,N1(C(c2cc(C)ns2)=O)CCCC2(CCN(C(=O)CCc3nnc(C)n3C)C2)C1 54013,C1(CNC(CSCC)=O)CCCCN1CC1CC1.c12ccc(cc1)CNC2=O 54014,C1(CNC(N2CC(CC)OC(C)C2)=O)CC2(CO1)CC1(C2)OCCO1 54015,C1(CC)CN(C(c2sc(CC(C)C)nc2C)=O)CCN1C(=O)C(C)C(C)(C)O 54016,S(=O)(=O)(CC(=O)NC(C(C)NC(=O)CCCNC(N)=O)C(C)C)NCC 54017,C1(N(C(CNC(CCOC)=O)=O)C)CC2CC1N(C(C1C3COCC13)=O)C2 54018,CN1CC(C(=O)NCC(C)(C)NC(=O)COC(F)F)c2ccccc2C1=O 54019,C1(NC(C2N(C)CC(F)C2)=O)CC12CCN(C(C1CCc3nn[nH]c3C1)=O)CC2 54020,N1(C(C(CC=C)C)=O)CCC2(CC1)CC2(CO)CNC(c1ccc(C)o1)=O 54021,C1(NC(c2c(F)ccnc2F)=O)CC1C1CCCN(C(=O)C2=C(Cl)CC2)C1 54022,N1(c2nc(OC)c(Br)cn2)CC2CCCC(C1)C2C(=O)NC(C)C1CC1 54023,C(=O)(C1=C(C)CCCC1(C)C)N(CC)CC1CCCN1C(=O)Cc1cccc(N)c1 54024,c1(NC(C(CC2CC2)NC(c2cnn(CCF)c2)=O)=O)cccc2c1CCC2 54025,Cc1nc(CNC(=O)CCC(=O)N(C)C)oc1C(=O)NC(c1nc[nH]n1)(C)C 54026,C1(CNC(C2(O)COC2)=O)CCC2(CCN(C(C3CC(C4CC4)=NO3)=O)CC2)O1 54027,Cc1cc(C(N2CC(F)(F)CC2CNC(=O)CCc2cnc[nH]2)=O)cc(N)c1O 54028,C1(NC(C(C)OCC=C)=O)C2CCC1N(C(c1nc(C)n(C)n1)=O)C2 54029,c1(NCC(=O)N(CCCNC(=O)C(C)(C)C2CCOC2)C)ncnc2[nH]cnc12 54030,N1(C(N2CCCC(S(C)(=O)=O)(F)C2)=O)CCOCCc2ccc(F)cc21 54031,C(C(=O)NNC(=O)c1ccccc1CC(F)(F)F)C1(C)CC1(F)F 54032,c1(C(=O)NCC2(C3CC3)CCN(C(C(COC)C)=O)C2)coc2ccc(F)cc12 54033,Cc1cccc(F)c1CC(=O)NC1(CCNC(=O)C(C)(C)CF)CC1 54034,C(C(C)CN=c1cc(C)nc(CO)[nH]1)NC(C=Cc1cccc(OCC)c1)=O 54035,c1(N(CC(CCC)N)CC)cccc(NC(=O)NCC)c1.C(COCC)O 54036,C1(CNC(C2CC(F)(F)C2)=O)CC2(CCC2)CN1C(c1cccn2nnnc12)=O 54037,CC12COC(C(N3CCC(O)(CNC(c4ccns4)=O)C3)=O)(C1)C2 54038,c1(N2C(CNC(C(CCC)OC)=O)C(C)CC2)ccc([N+](=O)[O-])cc1 54039,c1(CC(C(=O)OC)NC(c2ccc(O)c(Cl)n2)=O)cc(Br)ccc1I 54040,c1(C(=O)NC(C2(O)CCN(C(=O)CC3CC3)C2)C)nn(C)c2c1CS(=O)(=O)CC2 54041,Cc1nn(C)c(Cl)c1C(=O)NC12CC(CNC(c3ncccc3O)=O)(C1)OC2C 54042,N1(C(C(C)SCC)=O)CC2(CNC(c3[nH]c(O)nc3C)=O)CCC1CC2 54043,c1(C(C)NCC(COC)(C)C)ccc(C)c(C)c1 54044,c1(OC)cc(O)c(C(=O)NCCNC(C2CC2c2cccs2)=O)cc1S(N)(=O)=O 54045,C1(CNC(C2(C(N)=O)CCC2)=O)CC2COCC2N1C(=O)C(c1ccccc1)F 54046,Cc1c(C(N2CCN(CCNC(=O)C=CC(F)(F)F)CC2)=O)cnn1C1CCC1 54047,C(=O)(Nn1ccccc1=O)C1CC(NC(C(C2CC2)OC)=O)C1 54048,N1(C(C2C(C)CC2)=O)CC(C(N2CC(n3ccnc3)C2)=O)CC1(C)C 54049,C(C(N=[N+]=[N-])C(=O)N1CC(F)(CNC(=O)Cc2c(Cl)cccc2Cl)C1)OCC 54050,c1(C(=O)NC(C2CCCCC2)CNC(C(C)SC(C)C)=O)cccc(N(C)C)n1 54051,C1(C(N2CCC(NC(=O)Cc3ccc(Cl)s3)C(F)C2)=O)CN=C2N=CNN2C1 54052,N1(CC(COCC)O)CCOC(CNC(N)=O)C1 54053,C(CCCCCF)N(C(=O)C=CC(F)(F)F)CCOC 54054,Cc1cn2c(=O)c(C(N3CCC(CCNC(=O)C(C)P(C)(C)=O)C3)=O)cnc2s1 54055,Cc1nn(CCO)cc1C(N1CCC(N(C(=O)C(O)Cc2ccccc2)C)C1)=O 54056,c1(CC)cc(C(=O)NC(CC2CC2)Cc2ccccc2Br)cc(Cl)c1 54057,N1(C(c2cc(C)cc(C)c2C)=O)CCOC2(CCN(C(C3CCN3C)=O)C2)C1 54058,c1(C(=O)NC2CC(C)N(C(c3cc(Cl)n(C)n3)=O)C2)ccc2ncsc2c1 54059,c1(C(N2CCN(C(C3CCC(C)CC3)=O)CC2)=O)cc2cc(Cl)ccc2n1C 54060,c1(C(N2CC(C(C(N3C(C(=O)OC)C=CC3)=O)OC)C2)=O)ccnnc1C 54061,S(=O)(=O)(c1c[nH]c(C(=O)NCC(O)CNC(C2CC(C(F)F)C2)=O)c1)NC(C)C 54062,C(=O)(CCCCNC(=O)C(C)C1CCCO1)NCCSCCOC 54063,N1(C(C(CCC)C)=O)CCN(C(c2ccc[nH]2)=O)CC1c1cn[nH]c1 54064,N1(C(C(CSC)C)=O)CCC(C)(C(=O)NCc2cn(-c3ccccc3C)nn2)C1 54065,N1(C(c2cc(CC(C)C)on2)=O)CCN(C(=O)C=CC2CCC2)C(C)C1C 54066,C12(NC(Cc3ccc(C#C)cc3)=O)CCN(C(=O)CC(C)CCC)CCC1C2 54067,N1(C(C2C(C(C)C)C2)=O)CC(C)(CNC(c2onc3ccccc23)=O)CC1(C)C 54068,CC(C(=O)NCCCCCCNC(=O)CC(F)(F)Br)C(F)(F)C(F)F 54069,c1(OC)cncc(C(=O)NC2CCCC(C(N3CCC(F)CC3)=O)C2)c1 54070,C1(NC(C2C(OC)C2)=O)C2CC(O)C1N(C(=O)CNC(c1cscn1)=O)C2 54071,c1(NC(C2CN(c3ccncn3)CCO2)=O)ccc2c(=O)[nH]ccc2c1 54072,c1(C(N2C(CC(N3CCC(C#C)CC3)=O)CCC2)=O)cc(Br)c(O)c(Br)c1 54073,C1(NC(C(CC(C)C)(F)F)=O)CN(C(C2CC23CCCC3)=O)C2(CCCC2)C1 54074,C1(S(N)(=O)=O)(C(=O)NC(C)CN(C(=O)CCC#N)C)CCCC1 54075,CCCC(CNC(=O)CC1CC1C1CCC1)NC(C1(O)CCCC1)=O 54076,C1(=O)C(CN(C)C)N(C(C2CC2(F)Cl)=O)CC2CN1C2.CCOC 54077,N1(C(NC2CCc3cccnc32)=O)CC2(CCOCC2)c2ccccc21 54078,c1(C(C)NC(C(c2n[nH]c(C)n2)N(CC=C)CC#N)=O)ccccc1 54079,C(=O)(C1=CCCCO1)NC(C)CNC(C1(Oc2ccccc2)CC1)=O 54080,CCCCC(CNC(=O)CCOC(C)=O)NC(=O)CN1CCCCC1=O 54081,c1(C(=O)NCC23C(CN(C(C(n4ncc(C)c4)C)=O)C2)C3)c(F)cc(F)cc1Cl 54082,N1(C(C(c2ccc(Br)cc2)C)=O)CCC(F)C(NC(C2CS(=O)(=O)C2)=O)C1 54083,c1(C(=O)NC2CC(CNC(CC(CCC)O)=O)C2)cc(F)cc2nccnc12 54084,c1(C(C)NC(CC2N(C(CCC3C(C)C3)=O)CCC2)=O)ncc(F)cn1 54085,N1(C(c2c(CC)noc2)=O)CCN(C)C(C(=O)NCC2CCCCS2)C1 54086,O=C(C1Cc2c(Cl)cccc21)NCC1(F)CC(NC(c2c(F)cccc2F)=O)C1 54087,C(=O)(C(CCNC(=O)C(C1CC1)SC)OC)N(CCC)CC1CC1 54088,c1(C(N(CC(=O)NCC2(O)CCC(C)C2)CC#C)=O)cccc(CC)c1 54089,c1(C(=O)NC2CCC(N(C)C(c3ccccc3Cl)=O)CC2)cc(F)ccc1F 54090,c1(CN(CCNC(=O)NCC2CC(CC(C)C)OCC2)C)ccc(Cl)cc1Cl 54091,CC(C)CC(C(=O)NC1CCN(C(=O)C(C)OCCF)CC1)N1CCCCC1=O 54092,N1(C(CC(CN(C)C)(C)C)=O)CCC2(C=C(C(=O)NCc3ccc(O)nc3)C2)C1 54093,C1(C(N2C(CF)CC(OC)C2)=O)CC2CCC(C1)N2C(=O)Cc1cnns1 54094,N1(C(C(CCCC)O)=O)CCCC(C2CCCN(C(=O)CC3CC(OC)C3)C2)C1 54095,c1(C(=O)NCC2C(CNC(CCC(=C)Br)=O)C2)cc2ccccc2n1C 54096,N1(C(=O)CC2OCCO2)CC2CCN(C(C3CC(n4ccnc4)C3)=O)CC2C1 54097,C1(=O)CCCC(=O)O1.Cn1c(C(N2CCN(C(=O)CO)CC2)=O)nnc1S 54098,c1(CCC)onc(C)c1C(=O)NC(CNC(c1cc(C(F)F)ccn1)=O)C1CC1 54099,N1(C(C2(F)CC2)=O)CCC2(CC1)CC(NC(C13CCC(C(F)F)(CC1)C3)=O)C2 54100,c1(C(N2C(C)C(NC(=O)CC3CCC(=O)N3)CCC2)=O)ccc(F)c2[nH]ccc12 54101,C12(NC(CC(=C)C)=O)CCC(CNC(=O)CCCOc3ccccc3F)(C1)OC2 54102,c1(CC(=O)N(CCCC(C)C)Cc2ccc(C)s2)cn2ccccc2n1 54103,C1(NC(COCCCCC)=O)CCN(C(=O)CC(O)C(C)C)CC1O 54104,C(c1cn(C)cn1)=CC(=O)N(CCC(C)NC(=O)C(=Cc1c[nH]cn1)F)C 54105,C1(CNC(C2CN(C)C(=O)C2)=O)CC(C(=O)NCc2cn[nH]c2)=NO1 54106,CCCC1CC(=O)C2CC3C(C(Nc4cc(C)cnc4OC)C2C3)C(=O)N1 54107,CCCCCCC(C)NC(=O)CC1CN(C(c2csc(CC)n2)=O)C(C)(C)C1 54108,C1(C(N2CC(OC)CC2CSC)C(=O)NCCOC)CC2C=CC1CC2 54109,c1(-c2scc(C(C(=O)NCc3ccco3)N(CCC)C(C)C)n2)cccc(C)c1 54110,c1(CC)c(C(=O)N(C2CN(C(=O)Cc3ccn(C)c3)CC23CC3)C)cccc1C 54111,C1(CNC(CN(C(COC)=O)C)=O)CCC2(CN(C(c3c(C)n[nH]c3C)C)C2)O1 54112,N1(C(Cc2c(C)occ2)=O)CC(NC(c2cocc2C(N)=O)=O)CC(F)C1 54113,c1(C(CNC(=O)C(=O)N(C2C(CC)C2)C2CC2)F)ccc(F)cc1Br 54114,c1(C(N(C(CNC(C(C)O)=O)C2CC2)C)=O)ccn(CC(F)(F)F)c(=O)c1 54115,N1(C(c2cc(C)ns2)=O)CCCN(C(C2CCn3nccc3C2)=O)C(C)C1 54116,c1(C(N2CCN(C(c3cncc(C)n3)=O)C3C2C3)=O)ccc([N+](=O)[O-])cn1 54117,N1(CC(=O)NCC(C)N(C(c2c[nH]c(=N)s2)=O)CC)CCCCCC1 54118,N1(C(C2C(CNC(C(C)O)=O)CC2)=O)CC(C)c2ncccc21 54119,N1(C(CN2CCC(C)(O)C2)=O)CC2(CCCC(CNC(=O)C(F)(F)C3CC3)O2)C1 54120,N1(C(CC2ON=C(C)C2)=O)CCC(O)(CCNC(c2cc(C(F)F)cs2)=O)CC1 54121,CC(C)CCCCC(=O)NCCCC(O)C(=O)NCc1cc(Cl)ccn1 54122,C1(NC(CCN(CC=C)C(C2CC2Cl)=O)=O)C(O)CC1O 54123,c1(C(COC)NC(c2c(CC)ccs2)c2nnnn2CCCF)ccccc1Br 54124,c1(NC(C2CCCC2NC(=O)CNC(=O)C(F)(F)F)=O)cnncc1Cl 54125,C(=O)(CCCCCCCCN)N1CCN(CC(=O)Nc2c(OC)cccc2)CC1 54126,c1(CNC2CCC(NC(C3CCN(C(C)C)C3)=O)CC2)ccc(O)cc1O 54127,CC1(NC(C2CCCC2O)=O)CCN(C(=O)Cn2nnc(=N)[nH]2)C1 54128,C1(CNC(COCC)=O)CN(C(=O)C(C2CC2)SC)CCC1(C)C 54129,C1(C(=O)NC2CC(NC(c3n(CC)ccc3)=O)C2)Cc2cc(F)ccc2O1 54130,Cc1c(C(=O)NCC(C)CNC(=O)C(C(C)C)NS(C)(=O)=O)ccc2c1CCC2 54131,N1(C(CN2CC(CC)C2)=O)CCN(C(=O)CC2(OC)CC2)C2CC12 54132,c1(NC(C2(C)CN(Cc3cc(Cl)cnc3Cl)C2)=O)ccc(C(C)(C)C)cc1[N+](=O)[O-] 54133,C1(C(C)C(=O)N(c2ccn(C)n2)C2CC2)CCCN(C(c2cnc(=N)[nH]c2)=O)C1 54134,c1(CC(C)NC(c2cnn(C)c2C)c2n(CC)nnn2)cn(C)c2ccccc12 54135,C1(NC(c2c(CC)nn[nH]2)=O)CC(CNC(=O)CNC(=O)CN(C)C)C1(C)C 54136,N1(C(CCN(C(C)=O)C)=O)CCN(C(=O)C(Cl)=CCl)CCC1C 54137,C#CCC(C(=O)N(CC(C)COC)C)NC(c1cc(C2CC2)nn1C)=O 54138,c1(SC)cccc(F)c1C(=O)NCC1COCCN(C(c2cnccn2)=O)C1 54139,C1(CC(N2C(CNC(CC3C(=O)NC(=N)S3)=O)CC2)=O)CCC2(CC1)OCCO2 54140,c1(C(=O)NCCCCCNC(C2(C)CC2)=O)ccc(F)c(Cl)c1F 54141,c1(-c2cc(C(=O)NC(C3CC4(CCC4)C3)C)on2)ccccc1C#N 54142,C(=O)(N1OC2CCC1CC2)C1(C#C)CCNCC1 54143,Cc1cc(C(=O)NCC(C)N(C)C(C2CCCN2C)=O)ccc1C(F)(F)F 54144,CCCCC(CC)C(=O)NC1CCCC1NC(=O)C(C)(C)c1cnc[nH]1 54145,c1(C(CC)CC)cc(C(N2CCC(CN(C(=O)CCn3cnnn3)C)C2)=O)on1 54146,C=CCC(C)(O)C(=O)NCC1(OC)CCN(C(=O)C(C)NC=O)C1 54147,c1(CCCC(=O)NCC2CC2NC(=O)Cc2ccc(Cl)s2)nc2ccccc2s1 54148,c1(N2CCOCC(CNC(Cc3cccc(OC)n3)=O)C2)cc2nncn2cn1 54149,C1(NC(C2C(C)C2)=O)CN(C(=O)C(C)S(C)(=O)=O)CCC12CCC2 54150,CC1(C)CCC(C)(NC(C2(NC(c3sccc3F)=O)CC(CO)C2)=O)C1 54151,Cn1nc(CNC(=O)C(C2CCOC2)NC(=O)OC(C)(C)C)cc1C(F)(F)F 54152,N1(CC(=O)NCC(C2CCC2)NC(c2cccnc2O)=O)CCS(=O)(=O)CC1 54153,C(=O)(C1=CC(O)C(O)C(O)C1)N1C2CN(C(=O)Nc3cccc(C)c3)CC21 54154,C(C(C)C)(C(O)C(=O)NC(C(N1CC=CC1CN(C)C)=O)c1ccoc1)OC 54155,c1(C(N2CCCCC2CC(C)C)C(=O)NCC(=C)C)cn(CC(F)(F)F)nc1Br 54156,CCCCC(C(=O)NC1(C2CN(C(=O)C3=CCOC3)C2)CC1)N(C)C 54157,C1(CC(=O)N(C)CC2N(C(C(F)OC)=O)CCC2)CCCN(C(C)C)C1 54158,Cc1cccc(C(N2CC=CC(NC(C3CC(N=[N+]=[N-])C3)=O)C2)=O)c1F 54159,C(=O)(CCCC(C)(F)F)N(C1CCCN(C(C(C=CCCC)O)=O)C1)CC 54160,N1(C(=O)CCC2CCC2)C2CCC1CC(CNC(C1(N3CCOC3=O)CC1)=O)C2 54161,C(=O)(CC(C)(C)CC(F)(F)F)N1CCC(COC)(NC(=O)C(F)=C(C)C)C1 54162,C1(NC(c2cc(CC)n(CCO)n2)=O)CN(C(C2CC(=O)N(C)C2)=O)C(C)(C)C1 54163,N#CCCCC(=O)N1CC(F)CC1CNC(c1cccnc1C1CC1)=O 54164,c1(OC)c(Cl)ccc2[nH]c(C(N3CCCC(CNC(=O)C4=CCCS4)C3)=O)cc12 54165,C=CC1(CC(=O)NC2(C)CCN(C(c3c[nH]c(=N)nc3C)=O)C2)CCCCC1 54166,CCC(CO)CN=c1cc(C)c(S(=O)(=O)N2CCN(C)C(c3cccs3)C2)c[nH]1 54167,c1(C(N2CC(NC(C(C=C)(C)C)=O)C(C)C2)=O)c(C)ccn1C 54168,C1(C2CCC2)(CNC(C(CSC)OC)=O)CCN(C(c2ccncn2)=O)CC1 54169,N1(C(C2CN(C)C2)=O)CCC2(NC(=O)C3=COCCO3)CCCCC12 54170,N1(C(C2OCCN(CC)C2)=O)CC2(CCN(C(=O)CCC(C)C)CC2)CC1C 54171,CC1CCCCN1C(=O)CN(C(=O)C(=O)NC1CC1)CC1CC1 54172,N1(C(C(F)=CC)=O)CCN(C(=O)C(CC(F)F)c2ccc(F)cc2)C(CO)C1 54173,c1(CNC2C(c3c(C)n(C)nc3)OCC2)cc(C(F)(F)F)nc(C2CC2)n1 54174,C(C(C)C(C)C(=O)N1CCSCC1CCNC(=O)C(C)=C(C)C)OC 54175,C(=O)(CC(C)CC(C)C)NCCC(C(=O)NCCCOC=C)(C)C 54176,c1(CC)cc(C(=O)NC(c2cccc(C)c2)CNC(=O)C(C)OCC)ccc1Cl 54177,N1(C(C(=O)NCCNC(C)=O)=O)CCC(C)(C)C(CNC(=O)CC2CCCCO2)C1 54178,N1(C(C2(C)CCCO2)=O)CC2(NC(=O)CCC3(C#N)CCC3)CC1C2 54179,C=CCC(C(=O)NC1(CC(=O)NC(C)Cc2ccncc2)CC1)C(C)C 54180,c1(C(=O)NCC(CCNC(c2c(C)ccnc2C)=O)O)n[nH]c2cccnc12 54181,c1(SC)nc(=NC(C)C(c2ccccc2)NC(C2CCC(C)=C(C)C2)=O)s[nH]1 54182,C12(CNC(C(CC#C)(C)C)=O)CCCC(CN1C(=O)CNC(=O)OCC)C2 54183,C1(CC)CN(C(=O)Cc2ccc(C)s2)CC1C(=O)N(C)CC1(O)CCOC1 54184,C1(C(=O)NC(C(C)C)(C)CNC(=O)Cc2cnn(C(F)F)c2)CC2(CCC2)CO1 54185,C1(C(=O)NCC2N(C(c3c(OC)c(C)ncn3)=O)CCC2)CCCC1S(C)(=O)=O 54186,CC1COCCN1C(C1CC1(c1cccc(Br)c1)F)=O 54187,C1(NC(C2CC=CCO2)=O)CCOC12CCN(C(=O)Cc1ccccc1F)CC2 54188,C12(CNC(c3ccc(NC(C)=O)cc3)=O)CCCC1CN(C(c1cnn[nH]1)=O)C2 54189,C#CC1(C(N2CC(OC)CC(NC(c3cccc(F)c3C)=O)C2)=O)CCOCC1 54190,c1(OC)nc2ccc(CCC(N3CC(C)C3c3cccc(C)c3)=O)cc2[nH]1 54191,c1(C(N2CCCN(CCO)CC2)C(=O)NC)ccc(C(C)C)c([N+](=O)[O-])c1 54192,c1(CC(=O)NC(c2cnn(C)c2)C(=O)NCC(CSC)(C)C)ccc(C)c(C)c1 54193,N1(C(C2CCN(CC)C2)=O)CCN(C(=O)COc2ccc(F)cc2F)CC1CF 54194,N1(C(c2c(CC)c[nH]n2)=O)CC(O)CC1(C)C(=O)NCC(C)C(C)(F)F 54195,N1(C(C(CCC)(C)C)=O)CC2CCN(C(c3c(F)cc(Cl)cc3Br)=O)CC2C1 54196,C(=O)(C(O)CCS(C)=O)NCC(=C)CCNC(=O)CCCc1cccc(Cl)c1 54197,c1(N(CC(CC(C)C)OC)Cc2nnnn2-c2ccccc2Cl)ccc(-c2ccccc2)c(F)c1 54198,CC1(C)CCCC(CNS(=O)(=O)CC2(CF)CCOCC2)O1 54199,C1(NC(=O)C(O)CN2CCOCC2)CN(C(=O)CCOCC(F)(F)F)CC1F 54200,c1(N2CCC(c3scc(CC)n3)CC2)ccc(S(=O)(=O)N2CCC2C(C)C)cn1 54201,c1(C(=O)NC2C(CNC(C3N(C)CCC3)=O)COC2)cnc2c(c1)CNC(=O)N2 54202,c1(C(=O)NCCCN(C(C2CC23CCC3)=O)CC)scnc1C(F)F 54203,c1(CC)ccc(C(=O)N(C2(CC(=O)NCC3CC3(Cl)Cl)CC2)C)o1 54204,C1(CC(C)NC(c2cncc(F)c2)=O)CC2CCC(C1)N2C(C1CCCC1)=O 54205,N1(C(c2[nH]cc(OC)c(=O)c2)=O)CC2CCCC(C1)N(C(c1[nH]nnc1C)=O)C2 54206,c1(C2(C(N(C3CN(CC4(S(=O)(=O)N(C)C)CC4)C3)C)=O)CCC2)cccc(Br)c1 54207,O=C(C1=COCCO1)NCC1CC(F)CN1C(=O)CCCC1CCCC1 54208,Cc1nonc1C(=O)NC1(C(=O)NC2CSC2)CCSC1 54209,N1(C(CC2CC(OCC)C2)=O)CCC(C)C(CNC(c2ccc(O)nc2C)=O)C1 54210,C1(C(N2CC(OCCNC(C3CC=CCC3)=O)C2)=O)COCC1O 54211,C(=O)(C1=C(Cl)CCCC1)N(C(C)CN(C)C(c1ccsc1-n1cnnn1)=O)C 54212,c1(CN2C(C(=O)NCc3c(C(N)=O)nccn3)C(O)CC2)nc2ccccc2[nH]1 54213,C1(n2cc(COC3CC(C)C3)nn2)CCCN(C(C2CC(=C3CCC3)C2)=O)C1 54214,c1(N(C)C)ccc(F)c(C(=O)NC2CCN(C(=O)CCS(N)(=O)=O)CC2O)c1 54215,C1(C(N(CCC(C)NC(c2cnc(C(F)(F)F)s2)=O)C)=O)CCCOC1C(C)C 54216,C1(C(N(C(CNC(Cc2ccc(CC)cc2)=O)C)C)=O)CC12CCS(=O)(=O)CC2 54217,c1(CCC)cc(C(=O)NCCC(C)(C)NC(C2CCC2(OC)OC)=O)n[nH]1 54218,C1(CC(=O)NCCOCC(=O)NC)CN(C(=O)C(C)(C)C2CCOC2)CCO1 54219,C#CC1(O)CC(C(=O)NCCCOCCC(=O)NC(C(N)=O)C2CCCC2)C1 54220,C1(C(N(CCCNC(=O)CCc2nccs2)CC)=O)CNC(=O)CC12CCOC2 54221,c1(C(C)NC(c2cccc(Br)c2)c2nccn2C)ccc(F)c(F)c1F 54222,Cc1cn2cc(C(N3CCC(F)C(NC(c4ccc(O)cc4F)=O)C3)=O)sc2n1 54223,CCC(C)(C(=O)NCCCN(C(=O)C(F)(F)C1(OC)CCCC1)C)C(F)F 54224,N1(CC(=O)NCC(c2ccccc2)NC(=O)CCc2nccs2)CSCCSC1 54225,CCC(C)C(C(=O)N1CC(NC(C2C(C(C)N(C)C)C2)=O)C1)N(C)C 54226,C1(NC(C=CC=CCC)=O)C2CN(C(c3ccc(-c4ccc(F)cc4)[nH]3)=O)CC12 54227,CC1CN(C(=O)Cc2ccncc2OC(=O)C(C)(F)F)CC1Cc1ccccc1 54228,C#CC(C)(CC)NC(=O)C#CCNC(=O)C(n1nccc1C)C 54229,n1(CC(CC)O)cc(C(=O)NC2CCC(CNC(c3cnc(C)s3)=O)C2)nn1 54230,C#Cc1ccnc(C(N2CCC2CC(=O)N(C)Cc2cnn[nH]2)=O)c1 54231,S(=O)(=O)(c1ccc(C#N)cc1)NC(CC1(C)CN(CC2CNC(=O)C2)C1)=O 54232,N1(C(C2(C#N)CC(C#N)C2)=O)CCN(C(c2ccccc2)=O)CC(O)C1 54233,c1(C(=O)NC2CN(C(C(C3CCCOC3)OC)=O)C2)nonc1N 54234,C1(NC(=O)CC2CCC(F)(F)C2)CN(c2ccncc2[N+](=O)[O-])CCC12CCC2 54235,C1(CC)(CC)C(OC)CC1NC(=O)Cc1cccc(Sc2ccc(F)cc2)c1 54236,C1(F)(C(=O)NC(C2CN(Cc3c(OC(C)C)cccc3)C2)C)CCC(F)(F)CC1 54237,C(=O)(N=c1ccn(CCCO)[nH]1)C1N(C(c2ccc(COC)cc2)=O)CC(C)C1 54238,C1(C(=O)NC2CCC(Cn3cc(Cn4cccn4)nn3)CC2)(CC)CCCCO1 54239,N1(C(c2cnn(C)c2Cl)=O)C(C(N2CCC(N=[N+]=[N-])CC2)=O)C2CC(O)C1C2 54240,C(=O)(CC(CNC(c1c[nH]cc1C(C)C)=O)C1CCC1)NC(COC)CO 54241,c1(OC)ccc(NC(=O)N(C)CCN(C)C(=O)C2CC2)cc1Br 54242,C(=O)(C1=CCC(C)(C)CC1)NCC(CNC(c1c(C)c(C(N)=O)ccc1)=O)O 54243,C1(CNC(=O)CC2CC2)CC12CCN(C(c1ncc[nH]c1=O)=O)CC2 54244,C(=O)(C1CCCc2ncnn21)N1CCC(C(C)NC(=O)CC2=CCCCC2)CC1 54245,c1(NC(N2CC(OC3CCCCC3CC(F)(F)F)C2)=O)ccc(F)nc1 54246,c1(NC(C(n2cc(-c3cc(C)ncc3)nn2)C)=O)coc(S(C)(=O)=O)c1 54247,C1(NC(CNC(C(CC)C)=O)=O)CCCCN(C(C2(C)CC2C)=O)C1 54248,Cc1cc(C(N2CC3C(CNC(=O)CSC4CC4)C3C2)=O)c2sc(=N)[nH]c2n1 54249,CCC(C)CN(C)N(CCc1cccc(Cl)c1)CC 54250,N1(C(C(F)=CCC)=O)CCC(NC(C2CC(=C(F)F)C2)=O)C(F)C1 54251,c1(CCOCC(=O)NCCCN(C(=O)CC2C=CCCC2)C(C)C)ccccc1 54252,Cc1nn(CC(N2C3CCC(C3)C2CNC(C2CC(C)C2)=O)=O)cc1[N+](=O)[O-] 54253,C1(C(=O)NCC(C=C)O)CC(O)C(O)CC1CNC(C1CC(O)C(F)C1)=O 54254,CCC(CC(C)C)C(=O)N1CC2(C(=O)N(C(C)C(C)SC)C)CCC1CC2 54255,C(C)(CN=c1[nH]c2c(c(=NCCCN=c3cc[nH]c4ccccc34)[nH]1)CSC2)SC 54256,C(=O)(CCCCCO)NCCOC1(CNC(C2CC(C)OC2)=O)CCOCC1 54257,CCC(C)(C(=O)N1CCCC(COC)(NC(c2ccc(Cl)c(C)c2)=O)C1)C(F)F 54258,C1(C(N2CCC(NC(c3ccnn3C3CCC3)=O)(CF)C2)=O)CN2CCC1CC2 54259,c1(NCC(C)C)cc(N)ccc1-c1cccc(-c2nccn2C2CC2)c1 54260,N1(C(C(C=CC)O)=O)CCCC2(CCCCC2NC(c2cc(C)c(C)cn2)=O)C1 54261,c1(C(C)NC(c2n[nH]c(C)c2C(=O)O)=O)cc(Br)ccc1Cl 54262,c1(C(N2CC(N(C(C(Cc3c(C)nc[nH]3)O)=O)C)C2)=O)cc([N+](=O)[O-])cn1C 54263,N1(C(CCCC(C)=O)=O)CC2(CC(NC(=O)C(N3CCP(C)(=O)CC3)C)CO2)C1 54264,C1(NC(CN(C(CCOCCC)=O)C(C)C)=O)CCOC(CC)C1 54265,C1(C(N(C(CNC(C(CC(=O)OC)C)=O)C)C)=O)Cc2cccnc2C1 54266,c1(C(=O)OCC)nc(C)oc1OC.C12CC(C1)NC2=O.N12CCC1C2=O 54267,N1(C(CNC(=O)CN2CC3CC3C2)=O)CCC(Cn2cnnn2)C(O)C1 54268,c1(C(=O)NC(C(C)NC(C2(O)CCCCC2)=O)CO)ccc(Cl)c(C#N)c1 54269,CC(C(=O)N(CCCNC(=O)CCc1ncc(F)cn1)CCO)C(C)(F)F 54270,Cc1cc(C(=O)NCCN(C)C(c2cncc(C(F)(F)F)n2)=O)sc1Br 54271,N1(C(C(C2CC2)SC)=O)CC=C(C(=O)NC2CC(O)C2O)CC1 54272,N1(C(C(C)OC)=O)CCCN(C(c2cc(C)n(C(C)(C)C)n2)=O)C(C)C1 54273,CC(C)C(CC(=O)NC12CC(NC(c3ccnc(S)c3)=O)(C1)C2)C(C)C 54274,C1(N(C(=O)CCC2NC(=O)NC2=O)C)CCCN(C(=O)CCc2cnoc2)CC1 54275,O=C(CCN1C(=O)COc2ccccc21)Nc1ccc(OCC(F)(F)N)cn1 54276,c1(C(=O)NC(CC)CNC(=O)C(C2CC(F)(F)C2)OC)nn(C(F)F)cc1Cl 54277,c1(C(=O)NC(C2CCCCC2)CNC(C(C=C)(C)O)=O)nccc(C)c1F 54278,C1(C(=O)NCC2(O)CC(CNC(c3cc(COC)sc3)=O)C2)CC(=O)N(OC)C1 54279,N1(C(C23N(C(CCCN(C)C)=O)CCC2C3)=O)CCc2nnnn2CC1 54280,c1(NC(C2(C)CN(C(C(C)(C)OC)=O)C2)=O)csc2ccncc12 54281,c1(CC)ccc(C(N2CCN(C(=O)C3CC3)C3CC23)=O)cc1[N+](=O)[O-] 54282,c1(C(=O)NCC(CCNC(CCc2cn(C)nc2)=O)(C)C)c[nH]c2ncccc12 54283,C1(NC(CCC2C(C)C2)=O)CCN(C(c2ccc(OC(F)F)cn2)=O)C1(C)C 54284,N1(C(c2ccn(CC(F)F)n2)=O)CCN(C(c2cnc(O)o2)=O)C(C2CC2)C1 54285,c1(NC(COC)=O)cccc(NC(=O)NC(c2ccn(C)c2)C)c1 54286,c1(CC)cc(C(=O)NCC2CCC2NC(C2(Br)CC2(F)F)=O)n[nH]1 54287,CCCC(CC)CC(=O)NC1CCN(C(=O)C(c2ccc(C)cc2)C)C1 54288,C=C1CC(C(=O)N(C2CC(C)C2)C)(CNC(c2cc(Cl)cs2)=O)C1 54289,N1(CC(c2ccc(C)c(C)c2)C)CC(O)CCCCC1C(=O)O 54290,c1(NCCC(C)(C)SC)cc(C)c(S(=O)(=O)NC(c2ccncc2)CCO)cn1 54291,C#Cc1cccc(C(N2Cc3[nH]nc(C(N4CCC(C)C4(C)C)=O)c3C2)=O)c1C 54292,C1(CC(=O)NC2CONC2=O)OCC2CCN(C(=O)Cn3ccccc3=O)CC12 54293,CC(F)(F)C(F)C(=O)NCC1CN(C(=O)CSCC(F)F)CC12CC2 54294,c1(C(N2CCN(C(c3cc(C)nn3C)=O)CC(O)C2)=O)cc2cc(Cl)ccn2n1 54295,C#CCCC(O)C(=O)NC1COCCN(C(c2ncc(C(F)(F)F)cc2Cl)=O)C1 54296,C(CCCCN(C)C(c1c[nH]nc1-c1ccco1)=O)NC(C=CCN(C)C)=O 54297,N1(C(c2occ(C)c2)=O)CC(NC(=O)CC2CCC(=O)NC2=O)C2CCCC12 54298,C1(C(N(C2CCCCC2)C)=O)CC(O)CN1C(=O)CCc1csnn1 54299,C(C1CCCN1C(=O)CN1CCCCC1)=CC(N1CC(N(C)CC)C1)=O 54300,C(N=c1ccc(S(=O)(=O)NCc2ccc(F)c(Br)c2)c[nH]1)c1c(C)cccc1C 54301,C(c1ccc(F)cc1Cl)=CC(N1C(CC)CN(C(c2noc(C)c2C)=O)CC1)=O 54302,C1(N(CCC(=O)N2CC(N3CCCCC3)C2)C)CC1C1CC1 54303,c1(CNC(C(=O)OCC)Cc2ccccc2)cccc(CS(C)=O)c1 54304,N1(C(CC(C)C)C(=O)NCCN2CCOCC2)CC(C)(C)OC2(CCCOC2)C1 54305,c1(C(N2CC3(CN(C(CC(=O)NCC#C)=O)C3)C2)=O)cc(S(N)(=O)=O)cs1 54306,N1(C(CCC(CC)C)=O)CCCN(C(c2cnc(CC3CC3)s2)=O)CCC1 54307,N1(C(c2cc(CCC)n(C)n2)=O)CCC(C)C(NC(c2ocnc2CCC)=O)C1 54308,c1(-c2cc(C)c(OCCN)nc2)ccc2[nH]c(C(N3CCCC3CO)=O)nc2c1 54309,C1(C(=O)NCc2cnsc2)(CNC(CC(C)n2ccnc2)=O)CCCCC1 54310,C(=O)(C(F)CC(C)(C)NC(c1ccns1)=O)NC1CCN(C)C1=O 54311,c1(C(N2CCC(N(C(C3CC3c3cnc[nH]3)=O)CC)C2)=O)ccc(Cl)c(F)c1 54312,c1(OCC)ccc(F)c(C(=O)NC2CCCC2CNC(=O)COCCN(C)C)c1 54313,CCC(Cc1ccccc1)C(=O)N1CCNC(c2cccc(C(=O)OC)c2)C1 54314,Cc1ccnc(C2(NC(=O)N(C(C)CS(C)=O)C)CCC2)n1 54315,CC1CCC(NC(c2cc(Cl)no2)=O)CN1C(=O)C(N1CCN(C)CC1)C 54316,[N-]=[N+]=NCCCOCC(=O)NC(C(=O)NCCC(O)C1CCC1)C1CCC1 54317,C(=O)(CCCCC(=O)N1CCN(C(c2cccc(OC)c2)=O)CC1CO)OC 54318,CCCC(C)(O)CC(=O)N1CCCCC(NC(=O)Cc2nc(C(C)(C)C)cs2)C1 54319,N1(C(c2nnn(C)c2N)=O)CC2CCN(C(C3CCCOC3)=O)C2C1 54320,CCCCCC=CCC(=O)OCC(=O)NC1C(NC=O)CC1.C(C)(C)(C)OCC=C 54321,n1(CC(N2CC(N(C)C)C2)=O)cc(CNC(=O)C(O)C2CCCC2)nn1 54322,N1(C(N2CC(c3nc(C)on3)C2)=O)CCC2C(CCCN2C(=O)C2CC2)C1 54323,n1(CC(=O)N(CCC2CN(C(C)=O)C2)C(C)C)cc(C)cn1 54324,c1(CC(N2C(CNC(C3CC(=C4CC4)C3)=O)CC2)=O)ccc(O)c(F)c1 54325,C1(NC(COC(c2nccn2C)C)=O)CCN(C(c2occc2Br)=O)CC1F 54326,C1(N(C(=O)COCC2CCC2)CC#C)CCN(C(=O)Cc2csnn2)CC1 54327,C1(NC(CCCC=C)=O)CCN(C(C2CC3(CSC3)C2)=O)C(c2ccccc2)C1 54328,c1(Cc2nc(-c3cccc(C(C)O)c3)n(CC(F)F)n2)c(F)cccc1Cl 54329,C(CCCC(=O)NCC1C(C)CCN1C(=O)C1=CCOC1)N(C(C)C)C 54330,CC1CC2CC2CC1C(=O)NC1CCC(C)N(C(=O)CCC2CCCOC2)C1 54331,C1(N(C(CC(=O)NCC)=O)C)CS(=O)(=O)C12CCN(C(C1CCCCC1)=O)CC2 54332,N1(C(c2ccc(OC)o2)=O)CCN(C(=O)C(C)SC(C)C)C(c2cccnc2)C1 54333,C(=O)(C1=NOC2(CCC2)C1)NCC(CC)NC(=O)Cc1ccc(Cl)nc1F 54334,C(CCCCCCNC(c1ccco1)=O)n1cc(COCC)nn1 54335,C1(C(N2CCC(CC(C)NC(C(C=C)O)=O)CC2)=O)Cc2ccccc2C1 54336,c1(CC)cc(N)ccc1C(=O)NCC1CCC(NC(c2cnoc2C2CC2)=O)C1 54337,C(=O)(C(F)CC(C)(C)NC(=O)CC(C)(C)CN(C)C)Nc1c(CC)noc1 54338,C1(c2ccc(C)cc2)CC1N=c1[nH]c(=NCCC(C)O)[nH]c2c1COC2 54339,c1(C(=O)NCC2N(C(CCC(C)OCC)=O)CCC2)ccc(S(N)(=O)=O)cn1 54340,C1(C=O)CCN(S(C)(=O)=O)CC1.C12CC(F)CN1N(C)C2.C12(C=O)CCC1C2 54341,N1(C(COC(CC)C)=O)CCCCC(C2CN(C(c3cnc(OC)nc3)=O)C2)C1 54342,Cc1n[nH]c2cc(C(=O)NCC(C)NC(c3ncccc3Cl)=O)ncc12 54343,c1(N2CCC(N(C)C(C3(c4ccc(F)cn4)CC3)=O)C2)c(Cl)cncc1[N+](=O)[O-] 54344,CC1CCN(CCOC(C2(c3ccccc3)CC3(CC3)C2)=O)CC1 54345,c1(N(C)Cc2cc(C)on2)nc2c(c(=NCc3ncn(C4CC4)n3)[nH]1)CCC2 54346,Cc1cc(N2CC(F)(F)CC2CNC(C2CCC3CC3CC2)=O)ncc1C#N 54347,C1(C(=O)NC(CC(C)C)c2ccccc2)(CF)CCN(C(=O)OC(C)(C)C)CC1 54348,C1(OC)CN(C(=O)C(C)(C2CC2)N(C)C(C2COCC2(C)C)=O)CC12CC2 54349,C(=O)(C1CNc2ccccc21)NCCCCC(C)NC(C(C)OCC1CC1)=O 54350,N1(C(C(CCCNC(CC2CC(C)C2)=O)O)=O)CCc2c(F)cccc21 54351,N1(C(COC)=O)CCC2(CCC(C(=O)NCC3(N4CCOCC4)CCCC3)C2)C1 54352,N1(C(C2C(C)CCC2)=O)CCCC(CCNC(=O)COCC2CCOCC2)C1 54353,c1(CC(=O)NCC2(F)CN(C(=O)CC3CC(F)(F)C3)C2)cc(F)ccc1Cl 54354,c1(NC)ncccc1C(N1CC(NC(=O)Cc2ccsc2Cl)C(C)C1)=O 54355,C#CC1(C(=O)Nc2ccc(OC)nc2C)CCN(C(=O)C2=C(C)CC2)C1 54356,C1(Nc2cccn2CC)CC(NC(C2CCCC(C(=O)OCC)C2)=O)C12CCC2 54357,N1(C(C2C(C)C2C2CC2)=O)CC2CC3CC2C1C3NC(C1COCCO1)=O 54358,n1(C(C)C)ncc(C(=O)NCC(C2CC2)NC(C2(O)CC2)=O)n1 54359,c1(COCC(N2C3CC(NC(CSC)=O)C(C3)C2)=O)cn2cc(C)ccc2n1 54360,c1(C(=O)OC)cc2c(s1)CCC2NC(c1cncc(N)n1)=O 54361,CC1CN(C(=O)CCOCCNC(=O)CC#N)CC1CO 54362,C(C(C(=O)NCC12CCC(CC1)CC2)C(C)C)NC(C(C(C)C)OC)=O 54363,N1(C(C(C)SCC)=O)CC2(CNC(c3cc(Cl)nc(Cl)c3)=O)CC1CO2 54364,c1(C(=O)NCC(CNC(c2cccs2)=O)OC)cc2ccc(F)cc2o1 54365,c1(OC)ccc2[nH]c(C(=O)NCC3CCN(C(=O)CC(C)C)CC3C)c(C)c2c1 54366,N1(C(C(c2cnn(C)c2)C)=O)CC(NC(c2cc3sccc3s2)=O)CC(F)C1 54367,C1(CNC(COCC)=O)CCCN(C)C1C.C1CCC(=O)N1CC1CC1 54368,CC(C)CC(C(=O)NC(CC(C)(C)C)C(=O)N(C)Cc1ccnn1C)C(C)C 54369,C1(C(N2C(CNC(COCCOCC)=O)CC2)=O)CC(=O)N(CC(F)(F)F)C1 54370,c1(CNCc2c(C(=O)NCC(=O)Nc3ccco3)scc2)nc(C(F)(F)F)cs1 54371,C1(C(C)NCCCc2ccc(-c3ccc(F)cc3)s2)CCc2ncnn2C1 54372,CN1C(=O)CCC1CC(N1CC(O)CC1CNC(c1ccncc1N)=O)=O 54373,C1(NC(=O)C2CC2)CC2(CCN(C(C34CC(CO3)C4)=O)CC2)C1 54374,C1(C(=O)NC(CC(C)NC(=O)OCc2cccs2)C)CCN(C(=O)CCF)CC1 54375,c1(C(=O)NCC2CCC(NC(=O)C=Cc3ccncc3)C2)ccc2cncn2c1 54376,C1(O)(CNC(C(CC)(C)C)=O)CCCN(C(=O)CC2CCCC(C)(C)O2)CC1 54377,O=C(CCCC(F)(F)F)NC1CN(C(C2(CO)CC2(F)F)=O)CC12CC2 54378,C(C1=CCCN(C)C1)NC(C(C(C)NC(c1cnc(N)cn1)=O)C)=O 54379,C1(N(C(Cc2nc(C(C)C)sc2)=O)C)CCN(C(c2csc(=N)[nH]2)=O)CC12CC2 54380,N1(C(COCCCCC)=O)CCN(C(C2CCCN2CC(C)C)=O)C(C2CC2)C1 54381,CC1CC(C)N(C(c2nn3c(c2Br)CCC3)=O)CCN1C(=O)C1=CCCC1 54382,c1(NC2C(NC(C=C(C)Cl)=O)CS(=O)(=O)C2)ncnc2c([N+](=O)[O-])cccc12 54383,C1(c2nnnn2CCOC)(NCCOC(CC)(C)C)CCC(C(C)C)C1 54384,c1(C(CO)NC(C2(NC(COCC(=O)OC)=O)CC2)=O)cccnc1 54385,C(c1cn(C)nn1)=CC(=O)NC1(NC(=O)COc2cn[nH]c2)C(C)C1.C1C(=O)N1 54386,C=C(C)C1CCC(C)=CC1CC(=O)NC1(C)CN(C(c2ccc(Cl)cc2F)=O)C1 54387,C(=O)(C1=CC(c2ccc(F)cc2)=NS(=O)(=O)N1)N(CC(=O)OC)C 54388,C1(O)(CNC(C2CCC2)=O)CCN(Cc2cccc(-c3ccccc3)n2)CC1 54389,C=C=CCCC(=O)NC(C1CCN(C(c2cc(C)cs2)=O)C1)C 54390,N1(C(CN(C)C2CC2)=O)CCCC(C2N(C(c3cnc(O)s3)=O)CC2(C)C)C1 54391,n1(CC=C)cc(C(=O)NCC2(CC(=O)NCC3CC34CCC4)CC2)nn1 54392,Cc1ccc2c(C(=O)NCC(C)CNC(=O)CCc3ccc(F)nc3)coc2c1 54393,c1(C(=O)NCC(CC)NC(=O)C(F)=CC2CC2)ccc2c(c1)CCC2 54394,Cc1cc(C(=O)NCCN(C(=O)C=Cc2cc[nH]c2)C2CC2)cnc1C 54395,C(=O)(C(C)(F)C(C)(C)F)N1CC(CN(C)C(c2cn3ncccc3n2)=O)OCC1 54396,n1(CC)cc(Cl)c(C(=O)NCC2CCCN2C(c2sc(C)cc2C)=O)n1 54397,c1(C(=O)NCCCC2CCCN2Cc2sccc2Br)cc2ccccc2o1 54398,C(=O)(C(Cc1ccoc1)N(C)C)NCCC(C)NC(c1ccc(C(F)F)o1)=O 54399,C(=O)(CCCCC(=O)NC)NC12CCN(C(C(=O)NCCOC)=O)CC1C2 54400,CC(C)CC(C(=O)N1CCOCC1c1nncn1C)ONC(c1c[nH]c(Br)c1)=O 54401,C1(C(=O)NC(C)CC2(O)CCC2)C(CO)CCN1C(c1cnco1)=O 54402,N1(C(C2CC(CC)C2)=O)CCC2OCCN(C(c3ccn4cncc4c3)=O)C2C1 54403,CC1CC(C(N2CCCC2CNC(c2cccc(C3CC3)n2)=O)=O)CC(C)C1 54404,c1(C(=O)OC)c(C)cc(C)nc1NC(C)CC(C)NC(=O)CC(C)CC(C)C 54405,C1(NC(C(C)N(CC)CC)=O)CN(C(c2ncc(C(F)F)s2)=O)CCC1O 54406,C(c1cncc(F)c1)=CC(N1CC(C)C(NC(=O)CC2CCCCC2(F)F)C1)=O 54407,CC(C)C(C)(CNC(c1cnc(S)nc1)=O)NC(=O)C(c1ccc(Cl)s1)C 54408,c1(CCC(=O)NCC(C)(C2CCC2)NC(C(C)OCCCC)=O)c(C)n[nH]c1C 54409,c1(CC)cscc1C(=O)NCC(C)(O)CNC(c1c[nH]nc1C(C)C)=O 54410,C(CC(C)C)(C(=O)NC1CC2(C1)CC2NC(=O)CC1(CS(C)(=O)=O)CC1)OC 54411,C1(NC(c2cccc(OC)n2)=O)CC2(CCN(C(=O)C=Cc3ncc(C)[nH]3)C2)C1 54412,N1(C(C(C)SCCCC)=O)CCC(CNC(=O)C(CO)OC)C1C 54413,N1(c2nc(C)c(-c3ccccc3)nn2)CCCC2(CCCO2)CC1 54414,C(CN=C(NCc1ncc(C)s1)N1CCC2(CCCOC2)C1)N(C(=O)OC)C 54415,C(C1=CCN(C2CCC2)CC1)Oc1cncc(NC(C=CC(C)(C)SC)=O)c1 54416,C(=O)(C1CCCn2cnnc21)NC(CNC(c1ccc(CN(C)C)nc1)=O)(C)C 54417,C1(CNC(CCCC)=O)CC2CC2N1C(C1(c2ccccc2Cl)CCC1)=O 54418,Cc1nn(C)cc1C1CCCN1C(c1cnc(NCC2CC3CCC2O3)s1)=O 54419,c1(C(c2nnnn2CC(F)F)NC(c2c(C)n(C)nc2)C)nn(C)c2c1CCC2 54420,C(C(C)C)(C(O)C(=O)N1CCC(CF)(NC(=O)CN(CC(C)(C)C)C)C1)OC 54421,C1(C)(C(N(CCCC(=O)NCC(CC)(C)Cl)C)=O)CC(F)(F)C1 54422,C(=O)(C1=CC2CCC(C1)C2)N1CC(CCNC(C2CC3CC3C2)=O)C1 54423,C1(C)(CNC(C(C)NC(c2cc[nH]c2)=O)=O)CCCC1 54424,Cc1ncccc1C(=O)N(CCCNC(C12CC(O)C1C2)=O)C 54425,N12CC(C3CCCCC13)C2=O.C1(=O)C(O)C=CC(C)(C)N1.c1cnc[nH]1.C1(C)CC1 54426,CC1=C(CNC(=O)C(c2ccns2)NC(=O)OC(C)(C)C)S(=O)(=O)CCO1 54427,S(=O)(=O)(c1c(Cl)cc(Br)cc1Cl)N1CC(C)(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 54428,C12CC(C)(C1)NC2=O.C(=O)(C(N)=O)N(CCCOC)C 54429,N1(C(C2C(CCOC)C2)=O)CC23CCCC2(C1)CN(C(C1CCC(OC)C1)=O)C3 54430,C1(CC(N2CCCC23CCNC3)=O)CCN(S(=O)(=O)N2CCCC2)C1 54431,c1(C(=O)NCC2N(C(C(C(=O)OC)C)=O)CC(C)(C)C2)cccc2c1cnn2C 54432,C1(C)(C(N(CC(=O)NCC(c2ccccc2)O)C)=O)CC(C#N)C1 54433,c1(NC(C(=O)NC(CC=C)CO)=O)ccc(OC(F)(F)F)c(Cl)c1 54434,C(=O)(CC(F)(F)CNC(=O)OC(C)(C)C)NCc1c(OC)nccc1 54435,C(=O)(C(C)(C)C(N)=O)N1CCC(CN(C(c2c(NC)cncc2)=O)C)C1 54436,CCC(C)C(C)C(=O)NCCN(C)C(c1cnn(-c2cccc(Cl)c2)c1N)=O 54437,N1(C(CSCCCC)=O)CCC2CN(C(c3ccc(OC)nc3C)=O)CCC2C1 54438,c1(C(=O)OC)cccc(C(=O)NCC(C)(C)CNC(=O)CCF)c1C 54439,c1(SCC(=O)NCC2(NC(C(CC)N(C)C)=O)CCCC2)ccc(C)cc1 54440,CCC(C)(C)CCCC(=O)N1CC(NC(c2cnc(S)[nH]2)=O)C2(CC2)C1 54441,C1(n2nc(C(N(CC(C)CNC(=O)CCF)C)=O)c(O)c2)CCC(F)(F)CC1 54442,c1(C(c2nnnn2C(C)(C)CC)NCC(COCC)C)c(C)cc(Br)cc1C 54443,CCC(CNC(=O)CN1CCCS1(=O)=O)(CC)NC(C1C=CCCC1)=O 54444,CC(CNC(c1ccccc1O)=O)C(F)C(=O)NCc1c(F)cncc1F 54445,N1(C(C2(OC)CCC2)=O)CC2CCC(CNC(=O)CC3=CCCC3)C2C1 54446,CS(=O)(=O)CCC(=O)NC1CCN(C(c2csc(-c3cccnc3)n2)=O)C12CC2 54447,n1(CCC2C(C)CCN(C(=O)C(C)(C)CCCF)C2)cccc([N+](=O)[O-])c1=O 54448,CCCCCC(F)C(=O)NCCCN(C)C(C12CC(C)(C1)OC2(C)C)=O 54449,CC1(C)CC(CC(=O)NC2COCCC2NC(=O)CC2CC3(CC3)C2)CO1 54450,C1(C(=O)NCC2(NC(=O)Cn3cc(Br)cn3)CC2)CCC(=O)N2CCCC12 54451,Cc1coc2ccc(C(=O)N(CC(C)NC(c3cc(Cl)cc(F)c3F)=O)C)cc12 54452,c1(N(CCC)CC2(O)CCC2)nnc(COc2ccc(C)nc2)n1CCC#N 54453,N1(C(C2(F)CCN(C(c3cc(C)ncc3C)=O)CC2)=O)CCCC2C(O)CC12 54454,Cc1[nH]c2ncccc2c1C(N1CCOC(CNC(=O)C(O)CC(F)(F)F)C1)=O 54455,C1(CCOC)(NC(=O)C(C)Cc2cnco2)CCN(C(=O)CSS(C)(=O)=O)CC1 54456,C1(C(=O)N(CC(C)C)C)(CC)CCN(C(=O)CCC2CCOCC2)C1 54457,c1(C(N2CC(F)CC(NC(C(C)c3ccco3)=O)C2)=O)c(N)c(F)cc(F)c1F 54458,C(C(C)C)(C(O)C(=O)NC1CC(N(C(=O)CCc2cc(C)no2)C)C1)OC 54459,N1(C(c2ccn(CC)c2C)=O)CC(N(C(=O)CP(C)(C)=O)C)C2(CC2)C1 54460,C1(C)(C(N(CC=C)CCOC)=O)CN(C(C2CCC(C(N)=O)C2)=O)CC1C 54461,n1(CCC)nnnc1C(c1cc(C)[nH]n1)NCCc1cnoc1 54462,CC(CNC(=O)COCC1CC1)C(=O)NC(CO)CCC1CC1 54463,C1(C(N2CC(CC(=O)OC)C2)=O)C2CCC(C2)C1NC(=O)C(O)C(F)(F)F 54464,CCC(CC(=O)N1CC(=C(F)CNC(=O)CSC(F)(F)F)C1)C(F)F 54465,CCCC(CC)C(=O)N1CC2CC2(NC(c2cc(C(C)(C)C)c[nH]2)=O)C1 54466,C1(NC(CCSC)=O)CCN(C(c2ccc(CF)cc2)=O)CC1C 54467,C(=O)(C(CCCC(C)(F)F)N1CCC2C(CCCN2C(C)=O)C1)NCCOC 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54486,Cc1cc(C(=O)N(C2C3CN(C(C4CN(C)CCO4)=O)CC23)C)c(Cl)cc1F 54487,CC1Cc2ccccc2C1NC(=O)C(C(C)(C)C)NC(C1CN(C(=O)NC)C1)=O 54488,c1(C(=O)NC2N(C(C(C)Oc3ccc(C)cc3)=O)CC3CC32)cc(C#N)cn1C 54489,C1(C(N2CCN(C)C(=O)C2)=O)CC(C)(C)CCN1C(C1CN2CCC1CC2)=O 54490,N1(C(c2csc(Cl)c2)=O)CCC(=Cc2cccs2)CC1 54491,N1(C(C(C)NC(CC)=O)=O)CC2(CCN(C(c3cn(C)c(=O)cn3)=O)C2)C1 54492,C1(NC(COCCOCC#C)=O)(CF)CCN(C(c2c(C)ncn2C)=O)C1 54493,c1(C(=O)NCC(CNC(=O)CCc2ncco2)OC)cnc[nH]c1=N 54494,N1(C(c2c(CC)cc(Cl)cc2)=O)CCC12CCCN(C(=O)C(C)OC)C2 54495,C(=O)(NCC(=O)N(CCCC)CC)NCC(=O)NCC(=O)OC 54496,c1(-c2c(C(=O)NCCNC(C(COC)(C)OC)=O)cn(C)n2)cc(Cl)ccc1Cl 54497,CCC(C)C(O)CNC(=O)COC1CC(NC(C2(CC)CCCCO2)=O)C1 54498,N1(C(C2(OC)CC2)=O)CCOC(CCNC(N2CC(OCC)C2)=O)C1 54499,CC(C)CC(CC(C)C)C(=O)NCCC1CC(NC(c2cn(C)nn2)=O)C1 54500,c1(C(=O)NCCNC(c2c(C)cc(C)cc2O)=O)sc2[nH]c(C)nc(=O)c2c1C 54501,CC1(C(=O)NCCCC2CCCN2C(c2cnc[nH]2)=O)CCCC1(F)F 54502,C1(C(C)C)(C(=O)NCCCCN(C)C(c2coc(CC3CC3)n2)=O)CCCO1 54503,c1(CC)onc(C)c1C(=O)NCC(CC(C)C)NC(C1CCCN(C(C)=O)C1)=O 54504,C1(CC(=O)NC(C)C(C)NC(c2ccccn2)=O)CCCCC12CC2 54505,C1(C(NNc2cc(C)nc(C)n2)=O)CCN(S(=O)(=O)N2CCNCC2C)CC1 54506,Cc1[nH]nc2c1CC(C(N1CCCC(F)(CNC(=O)C(C)(C)C(F)F)C1)=O)CC2 54507,N1(C(CN2CC(C)(OC)C2)=O)CC=C(C(=O)NCC2CCN(C(N)=O)C2)CC1 54508,c1(C(=O)NCC(O)CCNC(C2(N(C)C)CC2)=O)cccc2[nH]ccc12 54509,c1(C(N2CC3C(NC(CCCCSC)=O)(CCC3)C2)=O)cccc(S(N)(=O)=O)c1 54510,N1(C(C2C(C)C2)=O)CC(C2CCN(C(=O)CC3CCCN(C(C)C)C3)CC2)C1 54511,c1(OC)csc(C(=O)NC2CCC(CNC(=O)CCCc3cccnc3)C2)c1 54512,CC#CCCCC(=O)NC(CNC(c1nnsc1C(F)F)=O)CC(C)C 54513,c1(C(=O)NCCCC2CCCN2C(C2CCC(F)(F)C2)=O)cccn2nncc12 54514,N1(C(C2CCC(C)(C)C2)=O)CCc2[nH]nc(CNC(C3CCOC3)=O)c2C1 54515,CC1CCc2onc(CNC(=O)CCC(C)c3ccccc3)c2C1 54516,c1(OC)cc(OC)nc(NC(CC2N(C(C3CCN(C)C(=O)C3)=O)CC2)=O)n1 54517,c1(CC(=O)NCCC2CCN(C(CCCc3onc(C)n3)=O)C2)cccc(F)c1 54518,N1(C(C(C)c2ccsc2)=O)CCOC(CN(C)C(C2(Cl)CCC2)=O)C1 54519,Cc1nn(C)c2c(N(C)CCn3cncn3)nc(=NC3CCCOC3)[nH]c12 54520,c1(OC)cncc(C(N2CC(CC(=O)NCC(C)OC(F)F)C(C)C2)=O)n1 54521,C(=O)(CC(C=C)CCC)NCC1CCCC(NC(CSCC#C)=O)C1 54522,C1(C(=O)Nc2c(C)ccnc2)CN(C(c2cccc(Cl)c2I)=O)CC(F)(F)C1 54523,C1(CC)CCCN(C(=NCCC2CC2)NCC(=O)N(C)OC)C1 54524,c1(C(N2CCCCC2CC=C)C(=O)NCC=C)ccccc1Br 54525,N1(C(C(CC)NC(N)=O)=O)CCCC(NC(c2sccc2Cl)=O)C1 54526,c1(C(=O)NCC(CC(C)C)NC(=O)CC2CN(C)C2)ccnc(C(F)(F)F)c1N 54527,Cc1[nH]c(C)c(C(=O)NCC(C)(C2CCC2)NC(=O)CCC(=O)N(C)CC)c1C 54528,N1(C(C(CCCC)F)=O)CCC2(CC(C(=O)N(C3CC(C(N)=O)C3)C)C2)C1 54529,N1(C(C(C=C)O)=O)CCCN(CCNC(=O)C(C)c2cncs2)CC1 54530,C1(NC(c2nc(C)sc2)=O)CCCN(C(=O)COC2CCCC(C)C2)C1C 54531,CCCC(CCC)CC(=O)N(C1CC2CC1N(C(c1ccc(F)c(C)c1)=O)C2)C 54532,N1(C(CSCCCC)=O)CC(C(=O)NCCNC2(N3CCCC3)CC2)CC(O)C1 54533,C1(C(=O)NCCN(C(C(CCCC)O)=O)C(C)C)Cc2nccnc2C1 54534,c1(C(=O)NC2CCC(N(C(=O)CN3CCCC3=O)C)C2)n[nH]c2c1CCSC2 54535,c1(N2CCC(=CC)C2)cc(C)c(S(=O)(=O)N2CCOC(c3ccccc3)C2)cn1 54536,C1(CNC(CN(CCOC)C)=O)(NC(=O)C(C)CO)Cc2ccccc2C1 54537,CC(C)CC(CNC(=O)CC1CC2(CCC2)C1)NC(=O)CCc1cccc(Cl)c1 54538,N1(C(C2CC(C)(C)C2)=O)CCN(C(C2CCC(C(F)(F)F)CC2)=O)CC(O)C1 54539,N1(CCC)C(=O)NC(c2ccc3nc(C4CC4)oc3c2)C(C(=O)OCC)=C1COC 54540,Cc1cccc(CCC(=O)N2CC(CN(C)C(C3CCCN(C)C3)=O)C2)c1 54541,N1(C(c2cn(CC=C)nc2)=O)CCC(N(C(=O)C(N2CCCCC2)C)C)C(C)C1 54542,N1(c2ncc(OC)cn2)CC(C(=O)O)C2(CN(C(C3CCNC(=O)C3)=O)C2)C1 54543,CC(C)C(CNC(C1CNC(=O)C1)=O)C(=O)NC1CCCCCC1CO 54544,c1(C(=O)NC2C(NC(C3C(OC)C3)=O)CCC2)csc2ccc(Br)cc12 54545,c1(C(c2nnnn2CCCSCC)NCCC(CC)C)nc(C)[nH]c1Br 54546,Cc1cc(C(=O)NCCOC2CCN(C(=O)CC(C)C)C2)c(C)n1C1CCOC1 54547,n1(C(C)C)ncc2c1CC(NC(=O)NC1CCCC1C(N)=O)CC2 54548,c1(OC)cc(OC)nc(C(=O)NC2CC3CC(NC(=O)C=C4CCC4)CC23)n1 54549,C1(CNC(=O)COCC2CCC2)COC(CNC(=O)CCOCC(F)F)C1 54550,N1(C(c2n[nH]c(CC)c2Cl)=O)CC(C)C(NC(=O)CN(S(=O)(=O)CC)C)C(C)C1 54551,c1(CC(=O)NCC2(COC)CCCN2C(=O)C(F)C(C)C)cc(C)ccc1C 54552,c1(C(=O)NC2CN(C(c3n(C=C)ncc3)=O)CC(F)C2)cccc(F)c1NC 54553,CCC(C)C(O)C(C)C(=O)N1CC(OC)CC1C(=O)NCc1ccc(F)c(Cl)c1 54554,S(=O)(=O)(c1ccsc1NS(=O)(=O)Cc1ccc(C(=O)O)cc1)NC(CC)C 54555,C(CCC)(C(=O)N1CCCC1C(N1CCCC1CCCC)=O)=CCC 54556,c1(CNC(C2C(=C)C2)=O)nc(CNC(C2COCCN2C)=O)cc(O)n1 54557,C1(CCC(=O)NC2CN(C(C(N)=O)=O)C2)CCC(=O)NC1 54558,c1(Nc2cncc(-c3ccc(C)cn3)c2)cc(N2CCCC2)nc(C)n1 54559,c1(-c2ccnc(NC(C(=O)OCC)=O)c2)ccc(O)c(C)c1C 54560,c1(N2C(C)CN(C(C3CC4CCC(C3)C4)=O)CC2)ncnc2c1cnn2C 54561,C#CCC(C(=O)NCc1nn(C)cc1C)NC(=O)CCCCN(C)C 54562,Cc1nc2ccc(C(N3CC(C(=O)Nc4nc5c(s4)COCC5)C3)=O)cc2[nH]1 54563,c1(C(=O)Nc2ccc(NC(COCC=C)=O)c(C)c2)c(C)[nH]c2ccccc12 54564,c1(C(=O)NC2CC3(C(NC(C(C)Cc4ccnn4C)=O)C3)C2)ccc(Cl)c(O)c1 54565,N1(C(c2cnc(SC)s2)=O)CC(NC(=O)CC2CC(C)(C)CO2)C2(CCCC2)C1 54566,c1(C(=O)NCC(C2CCOC2)NC(c2cnccn2)=O)ccn2ccccc12 54567,C1(C(=O)NC(CC)CNC(C2(CC)CCC(O)CC2)=O)CCC2C(C1)C2(F)F 54568,C1(n2cc(C(c3ccncc3)C)nn2)CCCN(C(=O)Nc2cncc(Cl)c2)C1 54569,CCC(CC)CC(F)C(=O)NC1C2CC3C1C3C2C(N1CC2(CCC(O)CC2)C1)=O 54570,C(C(C)CC(=O)NC1COCCC1NC(c1snc(Cl)c1Cl)=O)OC 54571,C1(C(=O)NCC2(COC)CN(C(C3CC=CC3)=O)C2)CNC(=O)CC1C 54572,N1(C(Cc2ccc(C)c(C)c2)=O)CCC2CN(C(=O)CC(C)(C)O)CC2C1 54573,N1(C(CC(C=C)C)=O)C2CCC1CC(O)(CNC(=O)CC1=CCCC1)C2 54574,c1(C(N(CCCNC(C2(C)CC2Br)=O)CC)=O)c[nH]cc1COC 54575,C1(C(F)(F)F)(C(N2CC(N(C(CN(CCC)C)=O)C)C2)=O)CCOCC1 54576,c1(CC(=O)NCC(C)(C)NC(C2CCC(C(=O)OC)C2)=O)cc(F)ccc1OC 54577,CC1(C)CN(C(=O)NC2CC(n3cncn3)C2)Cc2ccccc21 54578,c1(OCCC#C)ccc(CNC(C2CCNCC2C)=O)cc1 54579,C1(CC(=O)NCC2CN(C(c3c(C)snc3)=O)CC2C)CC(C)CC(C)(C)C1 54580,Cc1ccc(S(=O)(=O)NCC(N2CC3(C2)CN(C(C2CNC(=O)N2)=O)C3)=O)cc1 54581,C1(CC)CN(C(=O)COC2CCN(C)CC2)CCN1C(=O)C=C(C)c1ccco1 54582,C1(c2nnnn2C2CC(OC)C2)(NCCc2ccn(CC)n2)CCC1C1CCC1 54583,C12(C(N3CC(C)C(NC(c4cnn[nH]4)=O)C3)=O)CCC(C1)C2(C)C 54584,c1(OC)cc(CC(N2CCC(CNC(C3C(C)CC3C)=O)CC2)=O)ccn1 54585,C1(NC(c2cc(C)ncn2)=O)CC(C2CCN(C(c3cccc(C#N)c3)=O)C2)C1 54586,C1(CNC(=O)Cn2cccn2)COCCN(C(C2CC2OC(C)(C)C)=O)C1 54587,C12(C(N3CC(CNC(Cc4cncc(OCC)c4)=O)C3)=O)CCCN(CC1)C2 54588,C1(NC(CCOCC)=O)CC2C1CCN2C(c1ccc(C(C)(C)C)c(Cl)c1)=O 54589,N1(C(c2c(CC)cc[nH]2)=O)C(C(=O)NCc2snnc2C)CCC1C1CC1 54590,CON=CC(=O)NCCCCCNC(c1nnsc1N)=O 54591,C1(C(=O)NCCOC2CN(C(=O)C=CCF)C2)CC1C1CC(F)(F)C1 54592,c1(C(=O)NC(C2C3CCC(F)(F)C23)C(=O)OC)cc(C)cc(OC)c1C 54593,c1(C(N2C(C)(CC(N3CCOC4CC34)=O)CCC2)=O)c(Cl)cc(Cl)cc1Cl 54594,C1(C(=O)NCCCC(C)NC(=O)Cc2ccc(N)cc2)(COC)CCCCC1 54595,N1(C(c2cc(CC)on2)C(=O)NCC(F)F)CCC(NC(N)=O)CC1 54596,CC1(C)CC(=O)NC1CNC(C1OCCC1NC(=O)CN1CCCCC1=O)=O 54597,c1(C(=O)NCCCCN(C)C(C2(CO)CC2(F)F)=O)cc2cccn2cn1 54598,C(C(CO)CC(C)C)NC(C1(C)N(C(c2cc(C)sc2N)=O)CCC1)=O 54599,Cc1nc(NC(C)(CNC(C2(CC3CC3)CCCO2)=O)C2CC2)cc2nncn12 54600,C1(CNC(=O)CCc2cccs2)CCCN(C(C2CCC(F)(F)C2)=O)CC1 54601,c1(OCC(N2C(CNC(COC(C)(C)C)=O)CC2)=O)ccc(Br)cn1 54602,c1(C(=O)NCC(CN(C(=O)CC2COC(=O)N2)C)(C)C)cn2ccccc2n1 54603,N1(C(c2nn(CC)c(O)c2)=O)CC(NC(=O)CNC(c2ccsc2)=O)CCC1C 54604,Cc1cc[nH]c1C(=O)NCCCCc1cn(C2CCCC2N)nn1 54605,c1(CC)ccc(C(N2CCC(CNC(c3coc(Br)c3)=O)C(C)C2)=O)cc1N 54606,Cc1nc(C(=O)NC(C2CN(C(=O)C(C(C)C)NC(N)=O)C2)C)[nH]c1C 54607,S(=O)(=O)(c1cccc(=NCC2(F)CC2)[nH]1)NC1C(OC)C2(C1)CCC2 54608,C1(C)(CC)CC(NC(c2c(OC)cccc2C)=O)CN1C(c1cnoc1C)=O 54609,N1(C(c2c(C)n(C)cc2)=O)CCCC(C2CCCN(C(=O)CC(=O)N(C)C)C2)C1 54610,C12(NC(c3cc4oc(Cl)cc4[nH]3)=O)CCCN(C(c3cc(Cl)ccn3)=O)CC1C2 54611,c1(NC(C2CC(NCc3cnc(OC)s3)C2)=O)cnc2sccc2c1 54612,CC1COC2(CCC2)CN1C(=O)CSCCNC(=O)C(O)Cn1cncn1 54613,c1(SCC)cc(NC(=O)NCCOc2ccc(Cl)cc2Cl)ccc1OC 54614,C(=O)(C1=COCCO1)N1CC(OC2CCN(C(=O)CC3CC4CCC3C4)CC2)C1 54615,C1(C2CC2)(C(N(CC(C)NC(c2cc(C(N)=O)[nH]n2)=O)C)=O)CC=CC1 54616,c1(N(C2CNCCC2(F)F)C(c2ncccc2Cl)=O)ncnc2[nH]cc(I)c12 54617,CS(=O)(=O)CCC(=O)NCCC1(O)CCCN(C(C2CCC(C)CC2)=O)C1 54618,N#CC1(NC(c2cccc(F)n2)=O)CCN(C(c2ccc(Cl)nc2Cl)=O)C1 54619,c1(C(=O)NC(CCCCNC(C2(c3cc(C)no3)CC2)=O)C)occ2c1CCC2 54620,Cn1ncc2nc[nH]c(=NC3CC(C(=O)Nc4ncc(Br)cc4[N+](=O)[O-])C3)c12 54621,CC(C)(CCC(=O)N1CC(F)CC1C(N1CCC2(CC2)C1)=O)[N+](=O)[O-] 54622,CC1CCN(C(c2sccc2C2CC2)=O)CC1NC(c1nscc1Br)=O 54623,c1(C(=O)NCCC(=C)CNC(c2cnns2)=O)cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 54624,c1(N(CCC(N2CC(C(C)NC(=O)C(C)C3CCCC3)C2)=O)C)ccncc1 54625,C(C(C(=O)N(C)Cc1cccc(C)c1)C(C)(C)C)NC(C(C)=C1CC1)=O 54626,C(CC1CC1)(C(=O)NCCN1CC=CC1)NC(C1C(C)C1C)=O 54627,C(=O)(C(F)C(C)CC(C)(C)C)NCC1N(C(c2c(CC)occ2)=O)CC(C)(C)C1 54628,C(=O)(C1CCc2cccc(=O)n21)N1C(CNC(c2cn[nH]c2)=O)CCCCC1 54629,N12CC3C(C3C1)C2=O.c1(NCc2cnc(CC)s2)ccc(Cl)cn1 54630,N1(C(C23OCC(C(C)C)(C2)C3)=O)CCN(C(c2ccc(O)nc2)=O)C(C)C1 54631,c1(C(N(C(C)C)CC2CCSC2)=O)cccc(NCc2nccn2C)n1 54632,C1(C(N2CC(=C)C2)=O)CC2CCCC2N1C(C1CS(=O)(=O)C1)=O 54633,c1(C(=O)NC(CNC(Cc2nnc(C)s2)=O)C(C)C)c(Cl)cnn1C 54634,c1(CC)cc(C(=O)NCC(C)CNC(=O)CCCC2CCOCC2)ccn1 54635,c1(OC)cc(C(N2CCC(F)(C(=O)Nc3cn(C)nc3C)C2)=O)cc(OC)c1Br 54636,C(CC(=O)NC1CC(NC(C2(c3cccc(C)c3F)CC2)=O)C1)(C(F)(F)F)OC 54637,c1(CNC(=O)NCc2n(COC)ncc2)cccc([N+](=O)[O-])c1C 54638,C1(C(=O)NCC(C2CC2)NC(C2(c3cccs3)C(C)C2)=O)CCC(F)(F)CC1 54639,C=Cc1cncc(C(N2CCC(NC(c3ncncc3F)=O)C(F)C2)=O)c1 54640,C=Cc1ccc(C(=O)NC2CC2CNC(=O)Cn2nnc(-c3ccco3)n2)cc1 54641,c1(N2CC(OC)(CNC(=O)CCc3nc(C)cs3)C2)cc(=O)n(C(C)C)c(O)n1 54642,N1(C(c2cnc(OC)c(C)c2)=O)CC2(CCC(NCc3c(F)cccc3F)C2)C1 54643,c1(N(C(C2CS(=O)(=O)C2)=O)Cc2cccc(OC)c2)ccc(S(N)(=O)=O)cc1 54644,c1(OCC)nc(Cl)ccc1C(=O)NC1CCCN(C(C2CC3(CCC3O)C2)=O)C1 54645,c1(C(=O)NCCC(C)NC(=O)COCCN(C)C)cccc(OC(F)(F)F)c1F 54646,C12(C(N(CC(C)NC(C3CN(CCC)C(=O)C3)=O)C)=O)CCOC(C)(C1)C2 54647,C(=O)(CCCCC(=O)N1CCC(NC(=O)CCn2nc(C)c(C)c2C)C1)NC 54648,c1(C(N(CC(CNC(c2n(C=C)nnc2)=O)C)C)=O)cc(Br)ccc1O 54649,N1(C(=O)CC2CC2(Cl)Cl)Cc2ccccc2C(Nc2ncc([N+](=O)[O-])cc2Br)C1 54650,n1(CC)cnc(C(N2CC(NC(C3CCC(COC)C3)=O)C2)=O)c1 54651,C=CCC(C(=O)N(CCCNC(c1cc(F)ccc1C(F)(F)F)=O)CC)C(C)C 54652,Cc1ccc(CC(N2CC(NC(=O)Cc3ccsn3)C(O)C2)=O)cc1O 54653,Cc1cccc(C(=O)NCCC2CCC(NC(c3sccc3Br)=O)C2)c1 54654,N1(C(C2C(C)CCC2)=O)CCC2(CC1)CCN(C(=O)Cc1c(Cl)cccc1Cl)C2 54655,c1(OC)ccc(Cl)c(Cl)c1C(=O)NCC1CCN1C(=O)C(F)OC(F)(F)F 54656,O=C(C#CC1CC1)NCC1CC(F)CN1C(C1CCC1Cc1ccc(Cl)cc1)=O 54657,C1(C)(C(N2CC(OCC)(CNC(C3CSCC(=O)N3)=O)C2)=O)CCC(C)=C(C)C1 54658,N1(C(CC2CCN(C)C2)=O)CCN(C(c2cnoc2-c2ccco2)=O)CC(O)C1 54659,N1(CC(C)C)CCC(C(=O)NCC2CCCC2NC(=O)C2=CCOC2)CC1 54660,C1(NC(c2c(CC)cncc2)=O)CN(C(c2c(Cl)cncc2Cl)=O)CCC1C 54661,N1(C(c2ccc(OCC=C)cc2)=O)CCC(F)C(NCc2ccc(I)cc2)C1 54662,C(CC1=CCN(C(C2CCOC2C)=O)CC1)NC(c1cc(C)sc1)=O 54663,C=C1COCCN(C(=O)C=CC(C)NC(=O)CC(C)n2cccn2)C1 54664,O=C(CCCn1cncn1)NCCC1CCN(C(c2ccco2)=O)C1 54665,c1(C(=O)NCCCC2(NC(=O)COc3ccncc3)CC2)cnn(C2CC2)c1Cl 54666,C1(NC(C(C)Cn2ccnc2)=O)CC2(C1)CC2NC(=O)CCC(=O)c1ccc[nH]1 54667,C(C(=O)NC(CC(=O)N(C)Cc1cc(OC)no1)C1CC1)(C(C)C)OCC 54668,c1(C(=O)NCCC(=C)CNC(=O)CCC(F)F)cc2c(C3CC3)nn(C)c2s1 54669,c1(C(C)NC(C2(O)CCN(C(c3cnc(Br)o3)=O)C2)=O)ccc([N+](=O)[O-])cc1 54670,C1(C)(NC(c2n(CCC)nnn2)c2ccc(Br)o2)CCC2(CC1)CC2 54671,N1(C(C(CC(F)F)NC(C(CSC)OC)=O)=O)CCC(F)(F)C(F)C1 54672,N1(C(CN(CCC)C)=O)CCOCC1CN(C(=O)C(F)C(C)C)C 54673,S1(=O)(=O)c2cccnc2N1.CC1C(C)N(C)CCN1CCCN(C)C 54674,O=C(C1=CCCOC1)NCC1CC1CNC(C1C(C2CC2)C1(F)F)=O 54675,CCC(C#N)C(=O)N1CCC(C(=O)NCCCCO)(OC)C1 54676,c1(C(=O)NCC(CC(C)C)NC(C(C)(CO)NC(C)=O)=O)cnc2cc[nH]c2c1 54677,C1(C(=O)N)CCn2nnnc2C1.Cc1noc(C(C)C)n1 54678,C1(C(=O)NCCC2(NC(c3c(Cl)cn(C)n3)=O)CCCC2)CC12CC(F)(F)C2 54679,c1(C(=O)NC(C)(C)CCNC(=O)CC2(O)CCOC2)cc2ccncc2cc1F 54680,CC1(C)CCC(C(=O)NC2(CCF)CC2)CN1C(C1CN(C2COC2)C1)=O 54681,c1(NC(CC)CC(C)CO)ccc(S(=O)(=O)NCCc2csc(C)n2)cc1C#N 54682,C1(C(N2C(CCCNC(CN3C(C)CC3)=O)CCC2)=O)CN2CCC1CC2 54683,C1(NC(C2CN(C(N)=O)C2)=O)CN(C(c2ccc3n[nH]cc3n2)=O)CC2(CC2)C1 54684,N1(C(N(c2n(CC)cc(Cl)c2)Cc2ccccc2)=O)CCC2(C(C)(C)O)CCCC12 54685,C1(CC(=O)Nc2ncc(-c3ccccc3)cn2)CCCCC1NC1CCNC1=O 54686,O=S(=O)(c1ccc(=NCc2cccn3nnnc23)[nH]c1)NCC1(OC)CCC1 54687,C12(NC(c3ncn(CC)c3)=O)CC(CNC(=O)CCC(=O)OC)(C1)OC21CCC1 54688,C1(C(=O)NCCN(C)CCO)CC2(CCC2)CN1C(c1[nH]nnc1C1CC1)=O 54689,C1(=O)CS(=O)(=O)NCC2(CC2)N1.C=CCCC1(C(=O)N(C)C)CC1 54690,C(=O)(C(C#N)C(C)(C)C)NC(C(NOCC(=O)OC)=O)C 54691,c1(C(N(C(C)C)CCN(C)C(c2cc(Cl)cnn2)=O)=O)ccc2c(c1)N(C)CC2 54692,C1(C)(NC(C=Cc2occ(C)n2)=O)CCC(NC(=O)CC23COCC(C2)C3)CC1 54693,N1(C(c2cn(CCC)nc2)=O)CC2CCC(NC(c3oc(C)nc3C)=O)CC2C1 54694,N1(C(c2ccc(Cc3nn[nH]n3)o2)=O)CCOCC1c1cccnc1O 54695,C1(COC)CC(CNC(c2csc(=N)[nH]2)=O)N(C(c2[nH]c(O)nc2C)=O)C1 54696,C1(F)(C(=O)NCCCN(OC)C)CCN(C(c2cnc(C)nc2)=O)CC1 54697,CC1C(O)CC2CCC1N2C(=O)OC(C)(C)C.c1(C23CC(C2)N3)cccc(Br)c1 54698,c1(C(=O)OC)cc(C)nn1CC(=O)NC(C)CC(C)NC(=O)C(C)CC1CCC1 54699,c1(OCC(=O)NCC2N(C(c3c(C)n[nH]c3)=O)CCOC2)ccc(Cl)cc1Br 54700,c1(C(=O)NCC2N(C(C3N(C(N)=O)CC(O)C3)=O)CCC2)ccc(N)cc1Cl 54701,CON(C(=O)CCC1CCN(C(C2C(C)(C)C2(F)F)=O)C1)C1CCC1 54702,CCC(CC)(CO)C(=O)NC1CCN(C(=O)C(c2ccc(F)cc2)C)CC1 54703,C(C(C)C)(C(O)C(=O)N1CC(C(C(=O)NCC2CCOC2=O)OC)C1)OC 54704,C1(CN(C(CC(C)N2CCOCC2)=O)C)CCN(C(=O)C(C)(C)C#N)CC1 54705,C(C(C)(C)C(=O)NC1CCCC1CC(=O)NOCC=CCl)N(C)C 54706,c1(C(N2CC(C#C)(O)C2)C(=O)NCc2ccccc2Br)cc(F)c(F)c(Cl)c1F 54707,Cn1ncc(NCc2cccnc2P(C)(C)=O)c(Cl)c1=O 54708,c1(C(=O)NC2CCC(C)(CNC(c3n(C=C)ncc3)=O)C2)ccc(Cl)c(O)c1 54709,c1(C(=O)NC(CNC(CCC(C)OCC)=O)CO)cc(=O)n(C)cc1Br 54710,C1(C(N2C(C)(CC(=O)NC)CC2)=O)CC2(CC(NC(C3CCCC(=O)N3)=O)C2)C1 54711,C1(COCC)CCN(C(c2nonc2C)C(=O)NCc2ccccc2)C1 54712,N1(C(=O)NCc2ccn(C(C)C)n2)CCN(C2CCCOC2)CC1 54713,N1(C(Cc2ccc(C)s2)=O)CC=CCC1C(N1CCCC1CC1CC1)=O 54714,N1(C(CCCOC(C)=O)=O)CCCC2CN(C(=O)CSc3c(C)n[nH]c3C)CC12 54715,c1(CC(N2CCC(N3CCN(c4nncs4)CC3)C2)=O)ccccc1Cl 54716,c1(C(C(=O)NC2C(NC(Cc3c(C)scc3)=O)C2)C)ccc(F)cc1 54717,c1(C(=O)NC(C(C)C)C(C)NC(=O)Cc2cnc[nH]2)c[nH]c2c(C#N)cccc12 54718,C1(C(=O)NCC2CCC2)CC(OCC)C1.c12nc(n[nH]1)CCN2.C(C)(C)C.CF 54719,C1(CC)CCCCC1N(C(=O)C(C)(C)C1CCN(C(c2ccco2)=O)C1)C 54720,c1(C(=O)O)cc(CN2CC3(CC(C(=O)Nc4cc(O)nc(O)n4)C3)C2)cc(F)c1 54721,C(C(C)C(F)C(=O)NCCCC1CC(C)C1)NC(c1c(C)cc[nH]1)=O 54722,C(=O)(C(CC)(CC)CC)NC1CCC(C(=O)NC(CCC=C)C(=O)OC)CC1 54723,N1(C(C(C)c2ccco2)=O)CCCC(C)(N(C(=O)CCc2cccnc2)CCO)C1 54724,c1(CC(N2CC(CNC(c3cc(CCC)[nH]n3)=O)(COC)C2)=O)cnccc1C 54725,c1(C(N2CC(C)C(CNC(=O)Cc3csc(Cl)c3)C2)=O)cc(Cl)cc(F)c1N 54726,CC1CCCCC1CC(=O)NCC1(C)CC(C)(C)C1.C12CC(C1)NC2=O 54727,N1(C(C(CCSC)O)=O)CCOCC(C(=O)NCCC(C)SC)C1 54728,C(c1cccc(Cl)c1)=CC(=O)NCC1CCC(NC(c2cn(C)[nH]c2=N)=O)C1 54729,C1(CNC(C(C)=NOCC#N)=O)COC(C)(C)CN1C(=O)C1=CCCCO1 54730,n1(CCNc2ccc(NC(C(C)(C)C)=O)cc2)cc(C#N)ccc1=O 54731,c1(C(=O)NC2C(NC(c3nccc(C)n3)=O)COC2)ccc2cccnc2c1N 54732,N1(C(C2(C(=O)O)CCC(F)(F)CC2)=O)CCN(C2=NCCCN2)CC1 54733,C(C)(CCC(=O)N1CCC(C)(CCNC(c2cc(F)n(C)n2)=O)C1)SC 54734,C#CCCCC(C)C(=O)NCC(C(C)C)NC(=O)Cc1cccc(SC)c1 54735,C1(C(=O)NC2CC23CCN(C(c2cc(F)c[nH]2)=O)C3)CC12CCCCCC2 54736,N1(Cc2c(C)cccc2S(C)=O)C(=O)NC2(CCCCC2)C1=O 54737,C(=O)(NNC(=O)OCc1cccnc1)C1(NC(=O)OC(C)(C)C)CC1 54738,C1(SC)CN(C(C2CCC(N(C)C)CC2)=O)CC1NC(C1CC(C)N(C)C1)=O 54739,C1(NC(CCc2ccc(OC)c(OC)c2)=O)CCNC12CCOCC2 54740,N1(C(CSC)=O)CCC(C)(CNC(c2c(C)coc2C)=O)C1 54741,C(=O)(CN=c1cc[nH]cc1)N1C(CNC(C2C(C)(C)OCC2)=O)CCC1 54742,CC(C)C(O)C(C)C(=O)NC1CC2C(NC(c3ccc(F)cc3O)=O)C2C1 54743,CC1(O)COCCN(C(c2cc(CNC(=O)C(c3ccccc3)F)no2)=O)C1 54744,N1(C(CCC#CC)=O)CC(NC(C2(OC)CCOCC2)=O)C(C2CC2)C1 54745,Nc1c(C(=O)NC2CC(F)(CNC(C3CCN(C4CC4)CC3)=O)C2)cccc1Cl 54746,Cc1[nH]nc(Cl)c1NC(=O)N(C)Cc1cnn(C2CC2)c1C 54747,Cc1c([N+](=O)[O-])c(C(N2CC(NC(=O)C(=O)N(C)C)CC3(CC3)C2)=O)nn1C 54748,C1(CNC(=O)CCc2ccccn2)C(C2CC2)CCN1C(=O)Cn1cccn1 54749,c1(C(=O)NCC(CO)NC(CSCCC)=O)ccc(NC(=O)OC)c(C)c1 54750,C(=O)(C(=O)NNc1cc(C)c(Cl)cn1)Nc1c2ccc(C)cc2oc(=O)c1 54751,C1(C(=O)NCC(C)CNC(C2(C#N)CC2C(F)(F)F)=O)CCN(C(N)=O)C1 54752,C1(C2CC2)(CNC(c2ncc(Cl)cc2F)=O)CCN(C(C2(O)CCOCC2)=O)C1 54753,N1(C(c2ccc(N)c(C)c2C)=O)CCN(C(C23CCCCC2C3)=O)CC(C)(C)C1 54754,C(C(CC(=O)N1CC=CC1)NC(=O)C(C)CC#N)OC 54755,N1(C(c2cc(CCC)c(C)s2)=O)CC(NC(=O)CCNC(C)=O)C(C)(C)C1 54756,C1(c2cn(CC3CCN3C(C3CN(C4COC4)C3)=O)nn2)(N(C)C)CCCC1 54757,N1(C(C(CCC)CC)=O)CCCC2(C1)CN(C(C1(CCO)CC1)=O)C2 54758,C1(NC(C(CSC)O)=O)CC2CCC1CN(C(C1(F)CCCCC1)=O)C2 54759,c1(C(=O)NC(CC)CNC(=O)CCOC(C)=O)cnoc1CC(C)C 54760,N1(C(C(CCCNC(C2ON=C(C(C)C)C2)=O)O)=O)CCCN(C=O)CC1 54761,O=C1NC2(CCO1)CN(C(=O)CC1CCCC1NC(C1CCC=CCCC1)=O)C2 54762,C1(C)(C(=O)NC2(CC)CC2)CC(O)CN1C(=O)C(CC1CCC1)OC 54763,CN1CCCC(CNC(C2CC(NC(c3cc(F)n(C)n3)=O)C23CCC3)=O)C1=O 54764,C(=O)(C(C)(F)C(=O)OCC)N(CCNC(C1N(CCCC)CCOC1)=O)C 54765,C1(NC(c2cc(COC)sc2)=O)CN(C(c2n[nH]c(C)c2Br)=O)CC1C 54766,C(=O)(C(CO)C(C)(C)C)NCCC(C)(C)NC(CN(C)C(c1ccoc1)=O)=O 54767,c1(N2CC(O)(CNC(C(CCC)C)=O)C2)ncc(C)c(SCC)n1 54768,Cc1sc(CN2CCC(CC3(O)CC3)CC2)c(Br)c1C 54769,c1(OC)cc(C(C(=O)NC(C)(C)C)N(C2CCC(=O)NC2=O)C(C)C)cc(F)c1 54770,c1(C(C)C)nccc(C(=O)NC(c2cccc(Cl)c2)CNC(C2CC2C)=O)n1 54771,NS(=O)(=O)c1ccc(C(=O)Nc2ccc(Br)c(C(F)(F)F)n2)cc1 54772,c1(CN2CC(C(=O)Nc3cccc(O)c3Cl)OCC2)c(O)ccc2ccccc12 54773,c1(SC)nc(C(=O)N(CCCN(C)C(C2CC(F)CN2C)=O)C)c2ccccn12 54774,c1(C(N2C(C(C)NC(C3(C)CCC(=O)N3)=O)CCC2)=O)cc2nc[nH]c2cn1 54775,N1(C(CCOC)=O)CCC(NC(c2ccccc2N2CCCCC2)=O)C(C)C1 54776,C(C(C(=O)NC1CC(N(C)C(c2cnn(C)c2CC)=O)C1)C(C)(C)C)OCC=C 54777,N(C1CCCc2c(Br)cccc21)C(N1CC2(C1)CC2(F)Br)=O 54778,CC1(C)CCCC(NC(C2(C)CCN(C(c3nccnc3N)=O)C2)=O)C1 54779,c1(OC)cc(-c2csc(CO)c2)ccc1OC(F)F 54780,N1(C(c2cc(C)sc2)=O)CCN(C(c2cc(C3CC3)ns2)=O)CC1CCO 54781,C12(OC)CCC(NC(=O)CCC3CCN(C(C4(O)CCC4)=O)CC3)(CC1)C2 54782,C(=O)(CCC(=O)C1CC1)NC(C(C)NC(c1sccc1CN(C)C)=O)CO 54783,c1(C(N(CC(N2CCN(C(C(C)C(C)O)=O)CC2)=O)C)=O)cc(F)c(Cl)cc1Cl 54784,C1(NC(C)=O)CCCC(CC(=O)NC2CC2CNC(C23CC(C)(C2)C3)=O)C1 54785,c1(C(N2CC(NC(C3CCC(F)(F)CO3)=O)C2)=O)cnc2[nH]nc(O)c2c1 54786,c1(NCC(N2CC(c3c(CNC(C(CSC)O)=O)nco3)C2)=O)ccc(O)cc1 54787,c1(CCCSCCNC(=O)CN2CSCCSC2)ccc2ccccc2c1 54788,N1(C(C2(CC)CC2)=O)CCC2(CCN(C(c3cc(F)c4cn[nH]c4c3)=O)C2)C1 54789,c1(C(N(CC(CNC(C(C)OC(C)=O)=O)O)C)=O)ncc(C)cc1C 54790,c1(N(CCNC(=O)CC(C)C2CCCCC2)CC)ncnc(Cl)c1Br 54791,N1(CCn2c(C)ccc2C)CCCC(N(CC(c2ccccc2)O)C)CC1 54792,N1(Cc2ccn(CC)n2)CCC(NC(=O)CCC(=O)N2CCOCC2)CC(C)(C)C1 54793,C12(C(N3C(CCNC(Cc4nc(C)oc4)=O)CCC3)=O)CCC(F)(CC1)C2 54794,C1(C(N(C)CCNC(=O)CO)=O)C2CC3C(C2)C13 54795,c1(C(=O)NC2C3CN(C(Cc4nc(C)sc4)=O)CC2C3)c[nH]c2nccc-2c1 54796,C1(NCc2cnn(C)c2Cl)COC2(CCN(C(c3cnnn3C)=O)CC2)C1 54797,C1(CN(C)CCC2C(CC)CCCC2)CC12CCOCC2 54798,n1(CC=C)nnnc1C(c1csc(Br)n1)NC(c1nnc(CO)s1)C 54799,c1(C(=O)NCC2N(C(c3cc(C)c(N)cn3)=O)CC2)ccc(S(N)(=O)=O)cc1 54800,O=C(CS(=O)(=O)C1CC1)NC1COC2(C1)CN(C(c1cnc3cccnn13)=O)C2 54801,C1(F)(CNC(=O)CCC2CCCC2)CC(CN(C(C2(C3CC3)CCCO2)=O)CCC)C1 54802,Cc1nc(NCC2CCSC2)cc(=NCC(C(C)C)N2CCCC2)[nH]1 54803,C#CCCCCCNC(=O)C(CCC1CCC1)NC(C1CC1C(N)=O)=O 54804,S(=O)(=O)(c1ccc(NCCCCn2cnnc2)cc1Br)N(CCCC(=O)NC)C 54805,C(=O)(CCCCC(C)C)N(C1CCN(C(c2c(SC)nn(C)c2)=O)CC1C)C 54806,N1(CC(N2C(CCNC(CCC=CC)=O)CCC2)=O)C(C)CCC1C 54807,CC1(C)C(NC2CCC(C(=O)Nc3ccccc3)(CO)CC2)CS1(=O)=O 54808,C1(C(=O)NC(C)(C)CS(C)(=O)=O)CN(C(=O)CC2CCC(=O)NC2)CC12CC2 54809,CC1(C(=O)NC(c2ccccc2Br)CNC(C2CC2(F)F)=O)CC(F)(F)C1 54810,Cc1c(N2CCOCC2)ncnc1N1CCC(NC2COCC2C)CC1 54811,C1(C(=O)Nc2cccc(OC)c2)CCCN(C(=O)C=CCF)C1C 54812,C1(CNC(C2NC(=O)OC2)=O)(CNC(c2cccnn2)=O)CCCCC1 54813,c1(NC(C(CCCC)NC(C(=O)N)=O)=O)cn(CC2CC2)nc1C#N 54814,c1(C(N2CC(C(C)NC(c3cc(C)ns3)=O)C2)=O)c(C)ccnc1O 54815,c1(C(N2CCC(CC#N)C2)C(=O)OC)cccc(Cl)c1F 54816,S(=O)(=O)(CCC(=O)NCC1C=CC(NC(=O)C(c2ccccc2)F)C1)NC 54817,c1(CNC(c2c(CC)cc[nH]2)=O)ccc2c(c1)CCN(C(C1C=CCC1)=O)C2 54818,c1(NC(C2CC2C(N2C3COCC2C3)=O)=O)cnc(I)cn1 54819,N1(CCC)CCCC(C(=O)NC(C)CCNC(c2cc(CC)no2)=O)C1 54820,C(N=c1[nH]c(=NC2CCCC(F)(F)C2)c2ccccc2[nH]1)c1nc(C)c(C)[nH]1 54821,c1(C(=O)NCCC2N(C(CCC#CC)=O)CCC2)ccc2c(c1)OCCO2 54822,Cc1nc([N+](=O)[O-])cn1CCC(=O)NC1CC2CCC1CC2NC(=O)C(C)C 54823,c1(C(=O)OCC(=O)NC(c2ccc(F)cc2)C)cc2c(s1)CCCC2 54824,Cc1cn2c(CC(N3CCC(CNC(C4(C)C(C)(C)C4(C)C)=O)C3)=O)csc2n1 54825,c1(C(N2CCCC(C(C)NC(C(COC)NC(C)=O)=O)C2)=O)cnc(Cl)c(N)c1 54826,c1(C(N(C)CC2CCN(C(CCCC#CC)=O)C2)=O)cnc2c(c1)CCCC2 54827,C1(CNC(CCC(=O)N(C)C)=O)CC2CCCC2N1C(=O)CSCc1ncc[nH]1 54828,Cc1cc(C)c2[nH]c(C(=O)NC3CC(NC(C4CC4OC(C)(C)C)=O)C3)cc2c1 54829,c1(C(N(CCCNC(C2(O)CCC(CC)C2)=O)CC)=O)cccc2c1CC(=O)N2 54830,c1(C(=O)NCc2c(C(N3CCC(CC=C)C3)=O)con2)ccc(O)nn1 54831,C1(=CC(=O)NCCC2(O)CN(C(=O)C=CCCc3ccccc3)C2)CCSCC1 54832,c1(C(=O)Nc2nc(Cl)c(Br)cc2I)c[nH]c2cc(-c3cnn(C4CC4)c3)cnc12 54833,C1(NC(c2cc(CNC(C(CC)=CCCC)=O)no2)=O)CC(C)(C)OC1=O 54834,Cc1ncc(Cl)c(C(N2CCC(F)(CNC(=O)Cc3scnc3C)C2)=O)n1 54835,c1(C(=O)NC(C)CNC(c2cncn2-c2ccccc2)=O)c([N+](=O)[O-])cnn1C 54836,C1(C(=O)NC(CC)(C)CN(C)C(C2(C(C)=O)CC2C)=O)CC(C#N)(OC)C1 54837,Cn1cc([N+](=O)[O-])c(C(=O)NCCCCNC(c2cccc(C3CC3)c2Cl)=O)n1 54838,C1(C(N2CCC(C)C2CNC(c2cn(C)cc2C(F)(F)F)=O)=O)CC2(C1)CC2(F)F 54839,C1(C(N2CC(CN(C(c3c(OC)n[nH]c3)=O)C)OCC2)=O)OCCN(C)C1=O 54840,n1(CC(=O)NCCC2(O)CN(C(COCCCC)=O)C2)ncc2ncccc12 54841,c1(OC)c(F)cc(C(N2CCOCC2CNC(c2scnc2C)=O)=O)c(N)c1F 54842,c1(C(N2CCC3CN(C(COCC#C)=O)C3C2)=O)coc2c1C(=O)CCC2 54843,c1(C(N2CCC(C(C)NC(c3cc(CCO)on3)=O)CC2)=O)ccc(O)cc1Cl 54844,C1(C(N(C2CCCC(C)(C)C2)C)=O)CN(C(=O)C(F)n2ccnc2)CC(C)(C)C1 54845,c1(CC)ccc(C)c(NC(C2CCC(C)N2C(=O)CCC2CC2(F)F)=O)c1 54846,C(C(C)(F)C(C)(C)F)NC(C(CC1CCC1)NC(COC(CC)CC)=O)=O 54847,CCC(CC)N(C(=O)CCOCCO)C(C)CNC(=O)CSC(F)F 54848,C(N=c1[nH]c(N2CCCC3(CC2)CC(=O)N=N3)nc2cc[nH]c12)C1(C)CC(C)C1 54849,C(C1CCCN1C(=O)CC1CCSC1)=CC(=O)NC(C)C(C)(C)C 54850,c1(OCCC)ccc(CNC2(CC)CCNC2)cc1C 54851,C1(C(=O)NCC2(NC(=O)C(c3ccc(F)cc3)F)CC2)CC2CCCC(C1)C2 54852,N1(C(C2C(C)CCO2)=O)CCC(F)(C(=O)NC2(C)CCCC2O)C1 54853,Cn1cc(C=CC(N2CCC(C3CC3(F)F)C2)=O)c2ccccc12 54854,C1(CNC(c2ccc(F)cn2)=O)C(C2CC2)CCN1C(=O)COCC(F)F 54855,c1(C(=O)NC(CNC(C2(COC)CCC2)=O)CO)cc(OC)ccc1C 54856,C(C1c2ccsc2CCN1C(=O)COCC(C)C)NC(CCCCCCC=C)=O 54857,C12(CC3CCC(C1)O3)C(=O)OCCO2.C1CC(=O)C12CCCC2.C(=O)O 54858,C1(C(N2CC(CC(C(=O)NCC(C)C)F)C2)=O)CCCN(C(N)=O)C1 54859,Cc1c(C(=O)NCC2(CNC(C3CCCC(=O)N3C)=O)CC2)[nH]c2ccccc12 54860,C(=O)(C(O)CC(C)(C)C)NCC(C(=O)N1C(C(=O)OC)CCC1)C(C)C 54861,C1(CC(=O)NC(C)CC2CC2)CCN(C(C23C(=O)C4CC2C3C4)=O)C1(C)C 54862,C1(C(N2CC(O)(C(C)CNC(C3CCCC(F)(F)C3)=O)C2)=O)CCC(C)(C)CC1 54863,c1(C(N2CCC(N(CC#C)C(C3CCC3OC)=O)CC2)=O)cc2sc(C)cc2[nH]1 54864,c1(C(=O)NCC(C(=O)NCC(O)CN(C)C)N(C)C)ccc(C2CC2)cn1 54865,C(CC(=O)NC1CCCOC1)(C(F)F)NC(=O)CC1CC2(CCC2)C1 54866,Cc1csc(CC(=O)NC2(C(=O)NCc3ccnn3C)CC2C)c1 54867,N1(C(C2CC(=C)C2)=O)CCC(C(=O)NC2CC(C(F)(F)F)C2)(CF)C1 54868,C(=O)(CCCCC(C)CC)Nc1c(CC)cc(C(F)(F)F)cc1.N12CC(C1)C2=O 54869,c1(C(=O)NCC(CN(C(=O)C=CCN2CCCC2)C)O)cc2sc(Cl)cc2s1 54870,c1(C(N2CCC(C(CNC(C(CC)COC)=O)F)CC2)=O)ccc(C)nc1C 54871,c1(C(N2CC(O)(CNC(c3cc(Cl)cc(Cl)n3)=O)C2)=O)cc(Cl)cc(Cl)c1O 54872,c1(C(N(C(CNC(C=C(CCC)C)=O)C2CC2)C)=O)ccnn1CC 54873,c1(CC(=O)Nc2ccc(OCC(C)O)cc2)cc(F)ccc1Cl 54874,CC1(CNC(C2(CNC(=O)CC34CCCC3C4)CC2)=O)CCCCC1O 54875,c1(C(N2CCN(C(C3CCC(OC(F)F)CC3)=O)C3CC23)=O)nnc(O)cc1O 54876,Cc1c(C(N)=O)cccc1C(N1CC2(CCC2NC(C2C3CC4C(C3)C24)=O)C1)=O 54877,Cc1c(C(F)(F)C(N2CCCCC2C(C)NC(=O)C2=CCOC2)=O)cnn1C 54878,CCC(CC)C(C(=O)N1CCCCC1CNC(c1ccc(CCO)cc1)=O)OC 54879,CC(C)(C)CC(O)CC(=O)NC1CC2(C1)CC2C(=O)NC1(C(O)CO)CC1 54880,CCC(CC)(C(=O)NC1CCC(CNC(c2ccc(=O)n(CC)n2)=O)CC1)OC 54881,C1(CNC(CC=CCC)=O)(CO)CCCN(C(=O)C(F)C2CCC2)C1 54882,C1(OC(C)C(=O)NCc2ncoc2C2CN(C(=O)CNC=O)C2)CCCCCC1 54883,C1(CCC(N2C(CNC(c3c(C)coc3)=O)CCC2)=O)CCCCN1C 54884,CCC(C#N)C(=O)N1CC(F)CC1CNC(=O)C(C)(C)c1cccnc1 54885,N1(C(=O)CCOCC(F)F)CCC2(C1)CN(C(=O)C(c1ccccc1)O)CCO2 54886,n1(C(C)(C)C)cc(C(=O)NCC2CC2NC(C2CCC(C(F)(F)F)O2)=O)nn1 54887,N1(C(Cc2n(C)ccn2)=O)CCC2CN(C(C3OCC4CCCCC34)=O)C2C1 54888,Cc1cc(C(=O)NC2CCOCC2NC(c2ccn(C)n2)=O)ncc1C#N 54889,N1(C(CNc2nccc(OC)n2)=O)CCOCC(NC(=O)CCC2CC2(F)F)C1 54890,CCC(C)(CC)C(=O)NC(C1CCN(C(=O)C(=O)Nc2cccc(C)c2)CC1)C 54891,C1(NC(N2CC(COC)OC(C)(C)C2)=O)CCc2cc(OC)ccc2C1 54892,CCC(CCC(=O)N(CCC(=O)NC1CCN(C(C)C)CC1)C1CC1)OC 54893,c1(C(C)C)cc(C(=O)NC(c2ccccc2)C(=O)NC2CCCC2C(C)C)on1 54894,C1(NC(C23OCC(COC)(C2)C3)=O)CCCCN(C(=O)C(C(C)O)N(C)C)C1 54895,N1(C(CCc2ccc(C)nc2)=O)CCC2(CC(NC(C3(C)CCOCC3)=O)C2)C1 54896,c1(CC)nn(C)c(CNC(c2ncsc2Br)c2nnnn2C2CCC2)c1Cl 54897,N1(CCNC(C2CCSC2)=O)CCN(C(c2ncoc2C2CCCO2)=O)CC1 54898,C1(NC(c2cc(C(C)C)[nH]n2)=O)CC(F)(F)CC1NC(=O)C1=CCSC1 54899,Cc1cc(C(=O)NC2CCOC(C(=O)NCc3ccccc3CO)C2)n(C)n1 54900,O(NC(=O)CCCN(C(=O)C(C)CNC(N)=O)C(C)C)C(C=C)C 54901,c1(C(=O)NC2(CCCCNC(CC(CC)OC)=O)CC2)c(C)cccc1Cl 54902,N1(C(c2cccc(C#C)c2F)=O)CCC(NC(=O)CSCC)C(F)(F)CC1 54903,N1(C(C(C(=O)NC)(C)C)=O)CCN(C(=O)CCNC(C2CCCO2)=O)CC(O)C1 54904,CCCC(CC)CC(=O)N1CCN(C(c2c[nH]nc2C(C)(C)C)=O)CC1C 54905,C1(O)(CCNC(C(C)SC)=O)CCCN(C(c2[nH]c(=N)sc2C(F)(F)F)=O)C1 54906,C(N=c1nc2c(cnn2C)c(NCC(C)(F)F)[nH]1)C1(C(C)C)CC1 54907,N1(C(C2C(CC)CCO2)=O)CC(S(=O)(=O)N2CCN(C(C3CC3(F)F)=O)CC2)C1 54908,c1(C(=O)NCC(CC)NC(=O)C(F)NC(C)=O)ccc2c(c1)CCCN2C(C)=O 54909,N1(C2CCN(CCN(C)C)CC2)CCCC(C(N2CCCCC2C(N)=O)=O)CC1 54910,N1(C(COCC)=O)CCC(C2CCCCN2C(c2ccn(C3CCC3)n2)=O)CC1 54911,c1(C(=O)NC2CC(F)(CNC(C3CC(C)N(C)C3)=O)C2)cccc(S(N)(=O)=O)c1 54912,Cc1c(C(=O)N(CC(C)NC(=O)COc2ccc(OC)cc2)C)cc(O)cc1N 54913,C1(C(N(CC(N2CCC2C2CCCC2)=O)C(C)C)=O)CCCC(=O)N1 54914,C1(C(=O)OC)(CNC(C2N(C(CC3CC(=C)C3)=O)CC2)=O)CC=CC1 54915,C1(N(C(Cn2cc(-c3cccc(C)n3)nn2)=O)C)CCCCC1(C)C 54916,C1(CC(=O)N(C2CCCN(C(CC(=C)C)=O)C2)CC)OCCOC1(C)C 54917,n1(CC(=O)NC2CCN(C(C(C)CF)=O)CC2O)nc2n(c(=O)c1=O)CCOC2 54918,c1(C(=O)NCCSCC(=O)NC(C(CC)(F)F)(C)C)cc2ccccn2c1 54919,C(CNC(=O)Cc1csc(Cl)c1)(C(C)C(C)C)NC(Cc1cnc(C)[nH]1)=O 54920,C(=O)(CCCC(C)NC(N1CCOC(C(N)=O)C1)=O)OC(C)C 54921,c1(OCCOC)cccc2c(NC3CCC(C(F)F)CC3)c([N+](=O)[O-])cnc12.OCO 54922,N1(CC(=O)NC2C=CC(C(N3CCC3CO)=O)C2)C(=O)C=CC1=O 54923,C1(C(=O)NCCC(C)(C)NC(CC(C)c2cccnc2)=O)C(C)(C)C1(C)C 54924,C(C(C(C)C)NC(c1csc(S)n1)=O)(C1CCCC1)NC(CCOCCOC)=O 54925,C1(CNC(C(COC)(C)C)=O)CCN(C(=O)C(c2ccccc2Cl)C)C(C)C1 54926,C=Cc1cncc(C(N2CCN(C)C(C)C2)C(=O)NCCOCC)c1.C1COC1 54927,Cc1nsc(N)c1C(=O)NCC1(C)CCCN1C(=O)Cc1nc(C)c(C)[nH]1 54928,C1(NC(C(=Cc2cn[nH]c2)C)=O)CC(C)N(C(c2nnsc2N)=O)C1 54929,Fc1ccsc1C(c1cn[nH]c1)NCc1cccs1 54930,N1(C(C(n2cccc2C=O)C)=O)CCN(C(=O)C(C)NC=O)CC12CC2 54931,c1(NC(c2ccn(C)n2)C)nc(N2CCN(CC(F)(F)F)C(C)C2)nc2sccc12 54932,c1(C(N2CCN(C(C(C)SCC)=O)C(CCOC)C2)=O)cc2ccsc2c(O)n1 54933,CC(C(=O)NC1CC(CCn2cc(-c3ccncc3F)nn2)C1)C(F)F 54934,N1(C(C2N(C)CCC2)=O)CCCC2C1CCN2C(c1cc(Cl)ccc1[N+](=O)[O-])=O 54935,c1(NC)cc(Cl)ccc1C(=O)NCC12CC1CN(C(=O)CCCN=[N+]=[N-])C2 54936,C1(CC(=O)NC(C)CCNC(=O)CC2CCCCC2)NC(=O)CNC1=O 54937,N1(C(c2c(CC)nccn2)=O)CCCN(C(=O)C(O)Cn2cncn2)C(C)C1 54938,CCCC(C)(CCC)C(=O)NC1COCC1CNC(=O)C=Cc1ccoc1 54939,C(C1=CCCN(C)C1)NCC(=O)N(Cc1ccc(OCC)cc1)Cc1ccccc1 54940,CCC(CC(=O)N1CCC(CNC(=O)CCn2ccnc2C)C1)C1CCC1 54941,C(=O)(CC1=Cc2ccccc2C1)NC1CC(C)N(C(=O)Cc2n[nH]c(=N)s2)CC1 54942,C(CC1=CCN(C)CC1)N1CC(=O)N(C(C(N(OC)C)=O)C)C1=O 54943,C1(C(N(CCN(C(c2c(CC)nc[nH]2)=O)C)C(C)C)=O)C2CCCCCCC12 54944,CC1(C)CC(CNC(c2cnc(=N)[nH]c2)=O)N(C(=O)C(N)=O)C1 54945,C1(CNC(C(C)c2ccsc2)=O)CC2(CCC2)CN1C(=O)CC1CSCCS1 54946,C(=O)(C#CC1CCC1)NCC(CC=C)NC(=O)Cc1cccc(C(N)=O)c1 54947,C1(NC(C(C)O)=O)CN(C(c2nn(C)nc2Br)=O)CC1C(F)F 54948,N1(C(CN(c2ncccn2)C)=O)CCCC1C1CCCN1C(c1ccc(F)s1)=O 54949,N1(C(c2cc(C(=O)OCC)n[nH]2)C(=O)NC2CCCCC2)CC(C)CC(C)(C)C1 54950,CCC(C)(C(=O)NC1CC(C)N(C(=O)C(=O)NOC)C1)c1ccccc1 54951,Cc1onc(-c2ccccc2)c1C(=O)NCCn1cnc(C#N)n1 54952,C1(NC(CC(C(F)F)NC(C=CC(C)C)=O)=O)CCn2ncnc2C1 54953,c1(C(CC(=O)NCC(N2CCCS2(=O)=O)(C)C)O)ccc(O)c(O)c1 54954,c1(C(=O)NC(CCC)CNC(=O)C(F)CC2CCOC2)oc(C)nc1CC 54955,c1(C(=O)NC2CC(C)(NC(C3CN4CCN3CC4)=O)C2)cccc([N+](=O)[O-])c1N 54956,C1(C(N2CCC(N(C(Cc3ncc(CC)[nH]3)=O)C)CC2)=O)CCCCNC1=O 54957,N1(C(C2CC(N(C)CC)C2)=O)CC(O)CC1(C)C(=O)NCC(C)(C)C(C)(F)F 54958,C1(NC(C(CC)C#N)=O)(CO)CCCN(C(C2CC3CC(=O)C2O3)=O)C1 54959,c1(CSC)cn(C)nn1.C1(=O)C(CC2CC2)N1CC.C(=O)(CO)NCC(C)C 54960,C1(OC)(OC)CCN(C(C(=O)N2CCOCC2)C(C)C)C1 54961,N1(C(CCN(C(C)=O)C)=O)CC2CCCCC2(NC(=O)CSc2ccncc2)C1 54962,c1(CCC(=O)NCC(CNC(c2c(CC)occ2)=O)(C)F)cccc(F)c1 54963,C12(CC(N3CC(CC(C(=O)NC4C(OC)CCC4)F)C3)=O)CCC(CC1)C2 54964,C1(C(N(CCNC(=O)CSC2CC2)CC)=O)CC(=O)C1C 54965,Cn1cc(-n2cc(C3(O)CN(C(=O)CNC(c4ccc(Cl)s4)=O)C3)nn2)cn1 54966,C1(NC(C2C(C(C)C)C2)=O)CC2CCC1CN2C(C1CCC(C)CC1)=O 54967,c1(CC(=O)N(CC(C)NC(COCCC)=O)CC)ccc(C)nc1 54968,c1(C(N2C3CN(c4nccc(C)n4)C(CC3)C2)=O)cc(Br)c2ccccc2n1 54969,C(=O)(C1CN(C)C(=O)c2ccccc21)NC(C)CNC(=O)C=CCF 54970,c1(C(=O)NCCN(C(c2ccsn2)=O)CC2CC2)cncc(-n2ccnc2)n1 54971,C1(C2CCN(C(c3ccc(S(C)(=O)=O)o3)=O)C2)(NC(CS(CC)=O)=O)CC1 54972,C1(NC(C(C=C)(C)CC)=O)CC2CN(C(=O)C(CCC)C(C)C)CC2C1 54973,C(C1=NOC2COCC12)NC(C1(CC)CCCN(C(=O)Cc2csnc2C)C1)=O 54974,CCCCC(CC)C(=O)NC(C)(C)CNC(=O)CC1CCN1C(=O)OC(C)(C)C 54975,C(CNC(=O)CCc1c(C)n[nH]c1C)(C(C)(C)C)NC(C(C)OCCC#C)=O 54976,C12(CNC(c3c(Cl)cn(C)n3)=O)CCC(C1)N(C(C13CC(F)C1C3)=O)C2 54977,C(C(O)(C(F)(F)F)c1ccccc1)NC(CC(C)(C)c1ccccn1)=O 54978,N1(C(CCCC=C)=O)CCN(C(c2ccc(-c3ccccc3)[nH]2)=O)C(CCC)C1 54979,Cc1cccc(C(=O)NCC2(C)CCCN2C(=O)COc2ccccc2)c1F 54980,Cc1cc(C(N2CC(C(N3CCN(C)C(C4CC4)C3)=O)(C(C)C)C2)=O)nnc1C 54981,c1(C(N2CCCCC(CNC(c3cn(C)c(O)n3)=O)C2)=O)c(Cl)ccc(O)c1Cl 54982,C1(CC(C)C)CN(C(=O)CC(C)(C)C)CC1NC(=O)CC1C=NN(C)C1=O 54983,c1(OC)cc(C(=O)N(C2CCC(NC(c3[nH]ccc3C)=O)CC2)C)cc(F)n1 54984,CS(=O)(=O)c1cc(C(N2CCN(C(=O)C3=C(Cl)CC3)C(CCO)C2)=O)ccc1F 54985,c1(OC)c(Cl)cc(CN2CCC(O)C(C(=O)Nc3ncc(Br)nn3)C2)cc1Cl 54986,CCCC(CNC(c1cnn(C2CC2)c1)=O)C(=O)NCc1ncccc1O 54987,c1(CNC(CN(C(=O)C(COC)NC(C)=O)CC)=O)ccc(C)c(C)n1 54988,C(=O)(CCC(N)C(=O)O)N1CCN(Cc2c(OC)cccc2)CC1C 54989,Cc1ccc2c(c1)N(C(=O)NCCOC(C)(C)C)CCC2 54990,c1(C(=O)NCC(N(C(CCOC(C)C)=O)C)C2CC2)cc(Br)c2cccnn12 54991,N1(C(c2ccn(CC)c2C)=O)CCN(C(c2cnn3ccsc23)=O)C2CC12 54992,CC1CC(CNC(c2cc(CN(C)C)no2)=O)CN1C(=O)CCn1cncn1 54993,N1(C(c2cc(=N)[nH]c(=N)[nH]2)=O)C(CNC(=O)CC2C=CCCC2)CC2COCC12 54994,C1(C2CN(C(=O)CCc3nc(O)n[nH]3)C2)(NC(C2N(C)CC(O)C2)=O)CC1 54995,C(N=C(NCc1cc(C)on1)N1CCC2(C1)CC2(F)F)c1cc(C)nc(C)n1 54996,c1(NCC(=O)Nc2cccc3[nH]ccc23)cc(F)c(N2CCCCC2)c(F)c1 54997,C1(NC(COCCCC)=O)CC2CCC1N2C(=O)C(C(C)C)SC 54998,C1(NC(c2cnn(C3COC3)c2)=O)CC2CCC1N2C(=O)C(O)C1CCC1 54999,N(C1CCc2c(OC)cccc21)C(=O)NCc1c(C(=O)OC)sc2ccccc21 55000,CC(O)C(C(=O)NCC(C)(C)CNS(C)(=O)=O)N(C)C 55001,C1(CCC(=O)NC2C(C(=O)OC)CC2)CCCN1C(=O)CCCNC(C)=O 55002,CCS(=O)c1ccc(-c2ccc3c(C(=O)NCCCO)n[nH]c3c2)cc1 55003,C1(Nc2cccc(OCC#N)c2)CCCC2CNCCC12 55004,Cn1nccc1C1OCCC1NC(=O)NC(C12CC(CO1)C2)c1ccccc1 55005,C(=O)(C(C)CN(C)C(C)C)NC.c12nc(co1)N(C1CC1)C2=O 55006,C1(C(=O)NCC(C)NC(C(=O)NCC)=O)CCC(C)(C)CC1 55007,N(C(=NCCC1(C)OCCO1)NCc1cnccc1Cl)CC1(OC)CCC1 55008,CCC1=NOC(C(=O)NC(C)(C)CN(C)C(C2(C)CNC(=O)C2)=O)C1 55009,c1(NCC23C(CN(C(=O)OC(C)(C)C)C2)C3)nc(O)c2ncnc-2[nH]1 55010,C1(NC(c2cn(CC(C)C)nc2)=O)CCCCCN(C(=O)CC(C)F)C1 55011,CC1(C(=O)NCC2(F)CN(C(C3CC3CF)=O)C2)CC(c2ccccc2Cl)=NO1 55012,CC1(F)CC(C(=O)N(c2ccccc2)CCNC(=O)CCNC(=O)CO)C1 55013,CCC(F)(F)CC(=O)NCC1CN(C(=O)C(C2CCCCC2)N(C)C)CCCO1 55014,c1(C(N2CC(N(C)C)C(CNC(=O)CCC3CCCOC3)C2)=O)c(O)cccc1F 55015,C1(OCC(=O)NC(C)CC2CCCCN2C(=O)C2=CCCC2)CCCCC1C 55016,c1(C(=O)NCC(C)(C(C)C)NC(C(CCOC)C)=O)nc[nH]c2nccc1-2 55017,C1(C(=O)NCC2N(C(C(C(C)C)F)=O)CC2)C2(CCC2)C12CCC2 55018,CCCCCCCCC(=O)NCC1(OC)CN(C(C2(n3cncn3)CC2)=O)C1 55019,C1(CN(C(C2C(C(N(CC#C)C)=O)C2)=O)C)CCN(C(c2cnc(S)[nH]2)=O)CC1 55020,C1(CN(C(=O)Cc2cccnc2)C)CCCC1NC(C1CC(=C2CC2)C1)=O 55021,c1(NC(C(C(C)CNC(=O)CC2(C)CCC2)F)=O)cccc(N=[N+]=[N-])c1 55022,c1(C(=O)NCC(CC(C)C)(C)NC(C2CC=CC2)=O)cc2c(cn1)COCC2 55023,C(=O)(CCC1CCc2ccccc21)NCC(n1cc(C(C(C)C)O)nn1)C 55024,C#Cc1ccc(C(=O)NC(C)CN(C(=O)CS(=O)(=O)NCC2CCCO2)C)nc1 55025,C(=O)(CCC(C)(C)NC(c1nccn1CCN)=O)NCCCc1cn(C)nc1 55026,C(=O)(C(CO)C(F)(F)F)N1CCCC(CC(N2C(C)CC2)=O)CC1 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55063,n1(CCC)cc(C(=O)NC(c2cn(-c3ccc(Cl)cc3)nn2)C2CC2)c(C)n1 55064,c1(C(=O)NC(C2(O)CN(C(=O)C(F)CC3CCC3)C2)C)cccc(CS(C)=O)c1 55065,Cc1nn(C)c(C)c1CC(=O)NCC1C(C)CCCN1C(c1cnco1)=O 55066,c1(C(=O)NCCN(C(=O)C(C)c2cc[nH]n2)CCOC)nc(O)sc1C 55067,C1(C(N(CCCN(C)C(c2nnn(C)n2)=O)C)=O)CC2CCC1CC2 55068,c1(-c2cc(C(N(C)CC3(NC(C4CC5CC5C4)=O)CC3)=O)sn2)cccc(Cl)c1 55069,CC1C(OCc2ccccc2)CCCN1N(CCO)CCO 55070,Cc1snnc1C(=O)N(C)CCNC(=O)C(F)C1(NC(=O)OC(C)(C)C)CC1 55071,Cc1ccc(Br)nc1CNC(C1C2CCCC12)=O 55072,n1(CCOC)c(CSCCOC(C)CC#N)nc2c(C)cccc2c1=O 55073,c1(N(C)C(N)=O)ccc(N(Cc2cc(C3(O)CC3)[nH]n2)Cc2ccccc2)cc1 55074,N1(C(=O)C=Cc2ccco2)CCCC(C2CN(C(=O)C3=CC4CCCC34)C2)C1 55075,N1(C(C)=O)C(C)CN(CC(=O)NC2CC3(C2)CC3(F)F)CC1C 55076,N1(CC(=O)N(C2C3CN(C(CC(C)OC)=O)CC32)C)CCCCS1(=O)=O 55077,N1(C(c2cc(COC)cn2C)=O)CCC(N(C)C(c2nc(C)oc2C)=O)C(C)C1 55078,N1(C(CN2CCC(=O)CC2)=O)CC(NC(=O)CCc2cnn[nH]2)C(C2CC2)C1 55079,C(=O)(C(C1CN(C(c2cscn2)=O)C1)OC)N(CC(C)C)CC 55080,N1(CC(=O)NC2(C)CN(C(=O)CC3CCC(=O)O3)C2)CCC(F)(F)C1 55081,c1(C(C(=O)NCC2(CC(=O)NCCOCCC#C)CC2)F)ccccc1 55082,c1(OC(CC(=O)NCC(C2CC2)NC(CC)=O)C)cc(Cl)cc(Cl)c1 55083,N1(C(C(CC(C)(C)NC(C2OCCN(C)C2=O)=O)F)=O)CC2CCCC(O)C2C1 55084,c1(C(N2CCN(CC)C(C)C2)C(=O)NCC2CCOC2)ccc2c(n1)OCCO2 55085,c1(SCC(=O)N(CCCN(C(C2CN(S(CC)(=O)=O)C2)=O)C)C)ccccc1O 55086,CC(C)C(C(C)NC(=O)Cc1csc(-c2nc[nH]n2)n1)NC(=O)Cc1ccsc1 55087,N1(C(c2c(C(C)C)ccs2)=O)CC(NC(C2CN(C(N)=O)C2)=O)CC(F)C1 55088,C(=O)(C#CC1CCOC1)NC1C(NC(C2(OC)CCCC2)=O)CCC1 55089,C1(C)(CNC(CC(C)c2cnn(C)c2)=O)CCN(C(C2C(C)(C)C2(C)C)=O)CC1 55090,N1(C(C2CC(C(=O)OCC)C2(C)C)=O)CC(N2CCCC2)CC1C(=O)O 55091,N1(C(c2c(C(C)C)nns2)=O)CCC(OCCCNC(=O)C(F)C(C)C)CC1 55092,Cc1nc2n(n1)CC(C(=O)NCCCCC(C)NC(=O)CS(C)(=O)=O)CC2 55093,N1(C(c2cc(OC)c(C)c(OC)c2)=O)CC(C)(C)NC(=O)c2ccccc21 55094,c1(CNC(=O)NCC(CCCC)CCC)nc2c(C(F)(F)F)cccc2s1 55095,c1(C(N2CC3C(NC(c4ccc(C(=O)OC)cn4)=O)(C3)C2)=O)cc(C)c(C)cn1 55096,C1(NC(COC(C)(C)C)=O)CC2COCC(C1)N2C(=O)C(O)C1CC1 55097,C(C(=O)NCCN(C)C)(C(C)OC)NC(c1c(CC)ncs1)=O 55098,C(=O)(C(CO)C(F)(F)F)N1CCC2(C(C(=O)NCCc3n(C)nnc3)C2)C1 55099,c1(C(C)=O)c[nH]c(C(=O)NC(c2cn(C)nn2)C(=O)N(CCCF)C)c1 55100,N1(C(c2c(C)nco2)=O)CCC2(CCC2NC(C2CC23CCCCCC3)=O)CC1 55101,C(=O)(C(CC(F)F)C1CCC1)NCC(C)NC(c1nc(OC)oc1)=O 55102,C1(NC(=O)CCc2ccccc2)CCN(c2nc3ccccc3s2)CCC1CO 55103,c1(COC)nc(C(=O)NC2(CO)CN(C(=O)C(C)C3CCOC3)C2)co1 55104,C(=O)(C(O)CC(F)(F)F)N(CC)CC1CCCN(C(=O)CCn2cnnn2)C1 55105,C1(C(=O)NCC2C(C(=O)NCC3CC(O)C3)CC2)CCCC1F 55106,N1(C(COC2CC(NC(C(CCCC#C)C)=O)C2)=O)CCN2C(=O)OCC2C1 55107,C1(CNC(c2cc(C)c(C)o2)=O)CC2(C1)CC(C(=O)NCC1CC(O)CCO1)C2 55108,Cc1c(C(N2CCN(C(=O)CCc3ccoc3)C3CC23)=O)ccc2c1CCC2 55109,c1(CC(C)(C)C)cn(Cc2ncoc2CNC(c2ccc(F)s2)=O)nn1 55110,C1(CNC(c2c(C)onc2)=O)CN2CCCCC2CN1C(=O)C1=CCOCC1 55111,C1(NC(c2cc(C)oc2C)=O)CC(C)CN(C(C2(O)COC2)=O)C1 55112,c1(-c2cccc(OC)n2)cnn2c1CN(Cc1ccc(F)c(O)c1)CC2 55113,Cc1c(CC(N2CC3CC3(CNC(C3CCCC3(C)C)=O)C2)=O)ncn1C 55114,c1(C(=O)NC2C(C(=O)OC)CC2)cnc(C2CC2)nc1 55115,c1(CC)ccc(C(F)(F)C(N2CC(NC(c3cnc(O)n3C)=O)C(O)C2)=O)cc1 55116,C(=O)(C(C)(C)n1cc(NCc2ncnn2C2CCOCC2)cn1)OC 55117,C1(CCCN(C(=O)NC(C2CCCN2)C)CC2CC2)(C(F)(F)F)OCCO1 55118,N1(c2n(CC)c(COc3ccc(Br)cc3)nn2)CCc2cc(C)ccc2C1 55119,Cc1cccc(O)c1C(=O)NCC1(F)CC(CNC(=O)C=CCOC(C)(C)C)C1 55120,Cc1cc(C)c(S(=O)(=O)NS(=O)(=O)CCN2CC(NC(C)(C)C)CC2=O)cc1Br 55121,C=CCC(C)(C)CNC(=O)C(=O)NCC1CCOC1C 55122,Cc1cccc(CC(=O)N(CCCNC(=O)C(C)Cn2cccn2)C2CC2)c1Cl 55123,C12(CC(N3C(C)CC(CNC(C4(F)CCC4)=O)C3)=O)CC3CC(CC(C3)C1)C2 55124,Cc1cc(N2CCC3CN(C(=O)C(C)(C)N(C)C)CC3C2)ncc1[N+](=O)[O-] 55125,Cc1cc(Cl)cc(Cl)c1OCC(=O)N(C)CCNC(c1ncn(C)n1)=O 55126,C1(C(N2CCCC(NC(c3nc(CC)oc3)=O)(CO)C2)=O)CCCCCS1(=O)=O 55127,c1(C(=O)NC(CC)CNC(c2cc(N)cc(F)c2)=O)ncc([N+](=O)[O-])cc1Br 55128,N12CCC(C13CC3)C(=O)N(C)c1nsc2n1.C1(NC)OCCC1(C)C 55129,c1(CNC(=O)NCCC(=O)Nc2c(CC)cccc2)cc(Br)cnc1C 55130,Cc1cnc2n1C(C(=O)N1CC(CO)(NC(c3cc(=O)cc(Cl)[nH]3)=O)C1)CCC2 55131,Cc1cc(C(=O)N(C2CN(C(c3nnc(S)n3C)=O)C2)C)c2c(c1)CCO2 55132,C1(C(=O)NCCCCC=C)CCC2(CC2)N1C(=O)Cc1n[nH]c(C)n1 55133,CCC(CC)C(F)C(=O)N1CCCC1CC(=O)N(C1CN(C(C)C)C1)C 55134,CCCC(C(=O)N1CC(C)(OCC(=O)NCc2n[nH]cc2CC)C1)OC 55135,c1(C(=O)NC2(CNC(c3ccco3)=O)CCCC2)cn2c(n1)COCC2 55136,c1(Sc2cc(N3CC4CCC(CC4)C3)nc(C)n2)nc(Cl)nc2[nH]c(O)nc12 55137,N1(C(CCCNC(C(C)(C)C)=O)=O)CCCC(O)(CNC(=O)Cc2cncs2)C1 55138,c1(C(N2CC(O)CCC(NC(CC(COC)C)=O)C2)=O)ccc2c(c1)OCCN2 55139,C1(O)(CCNC(c2ccn(C(C)C)n2)=O)CCN(C(C2CCCCC2F)=O)CC1 55140,C=CC(C)CC(=O)NCC1CC(CNC(C2C=CCC2)=O)C1 55141,CC1(NC(=O)CSCCn2cncn2)CC(NC(c2csc(C3CC3)n2)=O)C1 55142,N1(C(COC(C)=O)=O)CCC2(CCN(C(=O)CN(C3CCSC3)C)C2)C1 55143,N1(C(CC(CNC(=O)CSC(F)F)OC)=O)CC2(CNC(=O)C2)C1 55144,c1(C(N(CC(CNC(Cc2nc(CC)sc2)=O)C)C)=O)cccc(NC(N)=O)c1 55145,C1(OCCC)CCCCC1C(=O)N(C)CCN1CCN(C(=O)CC(C)(F)F)CC1 55146,CC1CCCC(CC(=O)NCCCCNC(=O)C=C2CCN(C)CC2)C1 55147,CCCC(C(O)C(=O)NC(CC)(CC)C(C)C)NC(c1ccc2c[nH]nc2c1)=O 55148,c1(OC)cc(C#N)ccc1CN(CCC(C)C(=O)NCc1nnn(C)n1)C 55149,Cc1ccc([N+](=O)[O-])cc1C(N1CC2CC(NC(=O)Cc3scnc3C)C2C1)=O 55150,Cc1cccc2ncc(CN3CC(CO)C4(COC4)C3)n12 55151,N(C(=NCc1cc(-c2ccccc2)n[nH]1)N1CCCC(O)(CO)C1)CC(C)(C)C 55152,c1(C(=O)NC2CCC(N3CCOCC3)C2)ccnc(Cl)c1O 55153,Nc1ccc(CNC(Cc2cn(CC3(O)CCCCC3)nn2)CC(=O)O)cc1F 55154,C1(CNC(c2cnc3cc[nH]c3c2)=O)CN(C(C2CC2(Cl)Cl)=O)CCC1(F)F 55155,C12(C(=O)NC3CCCN(C(C4C5CC(F)(F)CC45)=O)C3)CCCCCC1OCC2 55156,c1(C(=O)NCCN(C(CCSCC)=O)C2CC2)cccc(F)c1 55157,C12(CNC(C3(C)CC=CCC3)=O)CCC(CNC(C3CC(F)(F)C3)=O)(CC1)CO2 55158,N1(C(CSCC)=O)CC2CCC(C1)N2C(=O)C=Cc1ccc(OC)c(C)c1 55159,C1(C(=O)NCC(C)CNC(=O)C(C)(C(F)F)c2ccccc2)CN2CCN1CC2 55160,CN1CCCC1CCCNC(C1(CC(F)F)CCNC1)=O 55161,N1(C(C2C(CC)C2)=O)CCC2(CCN(C(C3COC(C)C3)=O)C2)C1 55162,N1(C(C(C)OCC2CC2)=O)CCC(F)(CNC(=O)C(=Cc2cccnc2)F)C1 55163,N1(C(C(C)C)=O)CC(NC(=O)C(C)Oc2cccnc2)C(C#N)C1 55164,CCCCC(C)(CO)NC(C1CC=CC(NC(=O)CCc2cscn2)C1)=O 55165,c1(CC(=O)NC2CCC(CNC(C(=Cc3cnc[nH]3)C)=O)C2)cccc(Br)c1 55166,C1(C(=O)NCCC#C)CN(C(C2(CN(C)C)CC2)=O)CCO1 55167,C1(NC(C(CC=C)(C)C)=O)CC1C1CCCN(C(C2CCCC(O)C2)=O)C1 55168,c1(OC)c(CN2CCCC(C(=O)Nc3c(C)ncnc3C)CC2)cc(Cl)cc1Cl 55169,Cc1nncn1NC(=O)C1c2c[nH]nc2CN1C(=O)C1CCc2ccccc21 55170,c1(C(N)=O)ccc(C(F)(F)F)c(COC(=O)Cc2csc(NC=O)n2)c1 55171,C(=O)(CC(=O)N(C1CC(NC(C2(N(C)C)COC2)=O)C1)C)NCC#C 55172,C1(C(=O)NC(CCCC=C)C)N(C(c2ccnnc2C)=O)CCCC1(C)C 55173,CCC(C)(CO)C(=O)NCC(C1CCN(C(=O)C(C)SC(C)C)CC1)(C)C 55174,C1(F)(C(N2CCC(OCC(=O)N(CC(CC)O)CC)C2)=O)CCCCC1 55175,N1(C(c2nncc(OC)c2)=O)CC(NC(c2cc(C(F)F)[nH]n2)=O)CC12CCC2 55176,C12(C(N3CC(NC(C4CCCCCCC4)=O)C(O)C3)=O)CCN(CC1)S(=O)(=O)C2 55177,C1(NC(=O)C2=COCC2)CC(F)CN(C(c2ccc(=O)n(C3CC3)c2)=O)C1 55178,c1(C(=O)NC(C)CCNC(C2CC(C(C)(C)C)=NO2)=O)c(F)c(F)cc(F)c1F 55179,Nc1c(F)ccc(F)c1C(N1CCCCC(NC(C2CC3CC2C3)=O)C1)=O 55180,C#CCCCC(=O)NCCC1CSCCN1C(=O)COC(C)(C)CC 55181,CC1C(O)CCCN1C(c1n[nH]cc1CNC(c1ccc(=O)n(C)c1)=O)=O 55182,c1(C(=O)NC2C(CNC(CS(CC)(=O)=O)=O)CCCC2)cc2cccc(C)c2s1 55183,c1(C(N2Cc3[nH]nc(-c4ccnnc4)c3C2)=O)ccn2ncc(Br)c2n1 55184,C12(C(=O)Nc3ccc(C(=O)OC(F)(F)C(F)F)cc3)CCC(CO)(C1)OC2 55185,S(=O)(=O)(CC(C)C#N)N1CC(OC)OCC1 55186,c1(CC(=O)NC(CC)CNC(=O)CCC2CCC2)cccc(OC2CCOC2)c1 55187,N1(C(C(c2cccs2)SC)=O)CCCN(C(=O)COC(C)=O)CCC1 55188,c1(NC(C)C)cccc(C(N2CCC(CN(C(=O)CCc3cnc[nH]3)C)C2)=O)c1 55189,C1(C(N2CC(NC(C3CCN4CCCC4C3)=O)(CF)C2)=O)CCc2cnnn2C1 55190,CCC(C)(F)C(=O)N1CCCC(NC(=O)NC2CCCC2)C1 55191,C(=O)(C(O)CCCNC(=O)CC(C)N(C)C)NC(CC)C(C)(C)O 55192,C(=O)(CC(CC)c1ccco1)N(CCCCNCc1noc(C(C)C)n1)CC 55193,O=S(=O)(NCCc1c[nH]c2cc(F)c(Cl)cc12)N1CCC(F)(F)CC1 55194,CCCCC(C(=O)N1CC2CC1CN2C(c1n[nH]cc1Cl)=O)N1CCCS1(=O)=O 55195,CCCCCCCCC(=O)NCCOCCCNC(C1CCCCC1)=O 55196,C(=O)(C1=NOC2COCC12)NC(CNC(c1nn(CCCC)c(=O)cc1)=O)CC 55197,O=C1Cc2c(N3CCC3C(=O)Nc3ccc4nncn4c3)ncnc2N1 55198,c1(CNC(C2(C)CCN(C(C(CCC)OC)=O)C2)=O)cccc(F)c1F 55199,n1(C2CC(O)C2)nc(CN2CCCc3[nH]ccc3C2)c2c1CCCC2 55200,C1(CC(=O)NCCCCC2C(C)C2)(NC(C2CC3CCC3C2)=O)CCCCC1 55201,N1(C(c2ccn(C(C)C)n2)=O)CC2CN(C(c3ccnc(S)c3)=O)CC(C1)O2 55202,C1(C(=O)NCC2(F)CC(NC(C(C)=C3CCC3)=O)C2)CC2(CCCCC2)S1(=O)=O 55203,c1(C(=O)NCCN(C(CC(C)(C)OC)=O)CCOCCO)ccc(N)c(Cl)c1O 55204,C1(C(=O)Nc2c(C(=O)OC)csc2)CCN(C(c2cscc2OC)=O)CC1O 55205,C#CC1(C(=O)NCC2CCC(F)C2)CN(C(=O)CC2CC(N(C)C)C2)C1 55206,c1(C(=O)NCC2C(CNC(C3CCC(COC)C3)=O)C2)ccc(C(F)(F)F)nn1 55207,c1(C(=O)NC(CNC(c2onc(C)c2C)=O)C2CCC2)cc2c(nc1N)CCC2 55208,N1(C(C(COC)C)=O)CC2CCCC(C1)N2C(c1ccnnc1O)=O 55209,c1(CN2CCN(CCC(=O)NC3CN(C)C3)CC2)c[nH]c2cccc(F)c12 55210,N1(C(C(C2CCN(C(COCC=C)=O)C2)F)=O)CCC12CC(CO)C2 55211,c1(C(C)OC(=O)C(n2cc(C(c3ccccc3)O)nn2)C)ccc([N+](=O)[O-])cc1 55212,CCC(F)(F)C(C)(C)C(=O)N1CCC=C(C(=O)C(=O)C(N2CCNCC2)=O)C1.OC 55213,C(=O)(CCS(C)(=O)=O)N(C)CC1(NC(C2(C)CC3CC3C2)=O)CCCCC1 55214,c1(C(=O)NCC(CO)NC(C2CCS2(=O)=O)=O)ccn2c(C(F)(F)F)nnc2c1 55215,CC1CCN(C(C23CCCCC2C3)=O)C(C)C1NC(c1cn[nH]c1)=O 55216,N1(C(c2c(CC)non2)=O)CCC(NC(=O)C=C2CCCC2)C(F)C1 55217,CC(C)CCN=C(NCC(O)(C(F)(F)F)C1CCC(C)CC1)NC1CCCCC1 55218,C(=O)(C1=CC2CCC(C1)C2)N(C1CCC(NC(C(C(C)C)C)=O)CC1)C 55219,N1(C(Cc2cc(OC)no2)=O)CC(C)N(C(=O)Cc2cc(Cl)ccc2Cl)CC1C 55220,O=C(C1=CCCCC1)NC1C=CCC(C(=O)NCCCC(O)CO)C1 55221,C1(C(=O)NC(CC#C)CC)CNC(=O)CN1C(=O)C(COC)N(C)C 55222,CC(C(=O)NCCCC(=O)N1CC(O)(CO)C1)C(F)F 55223,C1(NC(CCCCC=C)=O)CN(C(=O)C=Cc2ncc(C)[nH]2)CC12CCC2 55224,N1(C(C(CC)CO)=O)CCC2(CC1)CC2n1cc(-c2ccc(N)cc2OC)nn1 55225,c1(C(N2CC(CNC(C3(C)CCOCC3)=O)C3C2C3)=O)ccc(Cl)nc1N 55226,C1(NC(C(CCC)NC(N)=O)=O)CCCN(c2nnc(C(N)=O)s2)CC1 55227,N1(C2CCN(C)C2=O)CC=C(CNC(C2CCCC(F)(F)C2)=O)CC1 55228,CC1(C(=O)NC2CC(CCNC(c3conc3C(C)(C)C)=O)C2)CCCCC1 55229,c1(C(=O)NCC2CCN(C(C(C)OC)=O)CC2)c(S(N)(=O)=O)ncn1C 55230,c1(COC(c2c(C)cccc2Br)=O)nc2ccccc2c(=O)n1C 55231,C(=O)(C(O)CNC(=O)C(C)CNC(C)=O)NCC1CC(C(=O)OC)C1 55232,c1(CC(=O)NCC(N(C(C(C(=O)NC)C)=O)C)C2CC2)ccc(C#N)cc1F 55233,c1(CCOC)nc(C(N2CCC(C(C)C(=O)N(C)C)CC2)=O)c(N)s1 55234,C(=O)(C(CO)C(C)(C)C)N1CCN(C(c2cc(SC)oc2)=O)CC1CO 55235,Nc1cc(F)cnc1C(=O)NCC(F)CNC(=O)CNC(c1ccsc1)=O 55236,c1(NCCOC)cccc(-c2cn(CC(C)NC(=O)CCCCC3CC3)nn2)c1 55237,N1(C(C=CC(=O)OCCCC)=O)CCC2CN(C(=O)CC3CC3C3CC3)CCC12 55238,c1(CN(C(C)CC2CC2)C)cc(-c2ccncc2)n[nH]1 55239,c1(CC)onc(C)c1C(=O)NCC1CC1NC(=O)C(N1C(=O)CCC1=O)C 55240,c1(C(C(=O)NC(C)C(=O)OC)N(C(C)(C)C)CC=C)cc([N+](=O)[O-])c(C)s1 55241,Cc1cc(C)c(C(=O)N(C2CCC2)C2CC2)cn1 55242,CCCC(C(=O)N1CCC(NC(c2cnoc2-c2ccco2)=O)C1)OC 55243,Cc1nc(C)n(CC(=O)NC2(CCNC(=O)Cc3sc(S)nc3C)CC2)n1 55244,c1(C(N(CCNC(C2CC3(CCO2)CC3)=O)CC)=O)cnc2ccncc2c1 55245,N1(NC(c2nncn2C)CC)CCC(C#N)(c2ccc(C)cc2)CC1 55246,c1(C(=O)NC2CCN(C(c3ccco3)=O)CC2O)cc2cnccc2o1 55247,CC1(C)CN(C(c2c(F)cc([N+](=O)[O-])cc2F)=O)c2cc(-c3ccsc3)cnc21 55248,CC(C)CC(C(=O)NCC1(NC(c2cccnn2)=O)CCCC1)C(N)=O 55249,N1(C(C2C(C(C)C)OCC2)=O)CC=CC(C(=O)NCCCC2(C)CC2)C1 55250,Cc1nscc1C(=O)NCCC1(C(=O)NCC(c2ccco2)O)CCC1 55251,c1(C(N2CC(NC(C(CC)O)=O)C2)=O)cccc2nccnc12 55252,c1(-n2c(CC3C(OC)COCC3)nc(C(C)C3CC3)n2)ccnc2ccsc12 55253,C1(CC)C(NC(c2ccn(C)c2C)=O)CCCN1C(c1ccc(=O)n(C)n1)=O 55254,C1(C(=O)NCCC2(NC(=O)C=CCO)CCC2)CNC(=O)N1 55255,c1(CN2CCC(F)(C(N3CCC(C#N)C3)=O)CC2)cnc2ncccn12 55256,C1(NC(c2c(Cl)cc(C)s2)=O)C2CC(CN(C(c3cc(CF)on3)=O)C2)C1CO 55257,C1(F)(CNC(C2(C)CC=CCO2)=O)CC2CCC(C1)N2C(c1cnc(C#N)s1)=O 55258,CCC(C)CC(=O)C(=O)N1CCCC(C(=O)NCC2(SC)CCC2)C1 55259,C(c1ccc(OC)cc1)=CC(N1CC(N(CC)CC)C1)=O.O(C(F)F)CCN 55260,c1(C(=O)NCC2(C)CCN(C(C(CCCOC)C)=O)CC2)ccc2occc2c1 55261,C(c1csc(S(=O)(=O)N2CCC2)c1)=CC(N1CC(C(=O)OC)C12CCOCC2)=O 55262,C(=O)(C1=C(C)OCCS1)N1CCC(CCOC)(NC(C2CCC2(F)F)=O)C1 55263,c1(OC)ccc2ccnc(C(C)NC(c3cc(F)ccc3C(=O)O)=O)c2c1 55264,C1(C(C)CO)CCN(c2cc(NCCN3CCC3)ncn2)CC1 55265,N1(C(c2cc(OCC)no2)=O)CCCCC1C(C)(C)CNC(c1cnsc1)=O 55266,CC1(C=CC(=O)NCC2(O)CCN(C(C3(C)CCC(=O)N3)=O)C2)CCOCC1 55267,Cc1ccc(CC(=O)NCC2(C)CCCN2C(=O)C=Cc2ccncn2)cc1C 55268,c1(C(=O)NC2CN(C(C(CC)O)=O)CC2C#N)c(Cl)ccc(OC)c1F 55269,C1(C)(CNC(C2CC(OC)C2)=O)CCN(C(c2cnns2)=O)CC1 55270,N1(C(c2n(CC)ccc2)=O)CC2CCCC2(NC(c2cccc3ccnn23)=O)C1 55271,CC(O)(C(=O)NCCCOCCNC(=O)CC1(C(F)F)CC1)C1CCC1 55272,C1(NC)CCOCC1NC(c1ncoc1CNC(C1(CF)CCOCC1)=O)=O 55273,c1(C(=O)NC(C)CCCNC(c2cnnn2C)=O)cnc2c(c1)CNC(=O)N2 55274,N1(C(C(CC)C)=O)CC(O)(C2(CNC(C3CCC(N(C)C)C3)=O)CC2)C1 55275,C(=O)(CCCCCF)N1CCC(NC(c2c(C)cc(CC)o2)=O)(COC)C1 55276,N1(C(C(CCCC)N(C)C)=O)CCCCCC(NC(=O)CC2CCC2)C1 55277,C1(CC=C)(NC(=O)C(C)CN(C)C(c2csnc2OC)=O)CCOC1 55278,N1(C(CCC=C=C)=O)CCCCC(CNC(C2CCCOC2)=O)C1 55279,C1(NC(c2n(COC)ncc2)=O)CCN(C(=O)CNS(=O)(=O)N(C)C)C12CCC2 55280,C1(NC(c2cn(CC)nn2)=O)CN(C(c2coc(C(N)=O)c2)=O)CC1O 55281,C12(C(=O)NCc3ncc(CC)[nH]3)CCC(NC(c3cnsc3)=O)(CC1)C2 55282,c1(C(C(=O)NCCC2CC(NC(C(C)(O)C3CCC3)=O)C2)O)ccc(Cl)c(F)c1 55283,c1(C(=O)NCCOCCN(C(C(C)SCC)=O)C)cc(Cl)c(C)cn1 55284,C=CCC(C(=O)N(CC(=O)NCC1CCC1)C1CCC1)NC(C)=O 55285,C(=O)(CC(CN(C)C)CC)N(C1CCC(NC(C2CCC(CC)O2)=O)CC1)C 55286,C(=O)(C#CC1CCCCC1)N1CCC2(CN(C(C(C(C)C)F)=O)C2)C1 55287,c1(C(NNC(C(=O)OC(C)(C)C)=O)=O)nc(=NCc2ccco2)[nH]cc1Cl 55288,C(C1OCCc2ccccc21)NC(NCc1nc(OC)c(C)s1)=NCC1CCC1 55289,Cc1nn(CC(=O)N(C(CNC(C2(Cl)CC2(F)F)=O)C2CC2)C)cc1[N+](=O)[O-] 55290,c1(NC(C2N(C(CC(C)O)=O)CC(C)C2)=O)cc(Br)cc(F)c1C#N 55291,Cc1nc(Cl)ccc1CC(=O)NC(C)C(C)(C)NC(c1ncoc1C)=O 55292,C(=O)(C1=CNC2=NCCC2=C1)NCC1(C)CCCN(C(Cn2c(C)cnc2)=O)C1 55293,c1(CNCC2OCCN(C(C3N(C)CCC3)=O)C2)ccc(Br)cc1C#N 55294,S(=O)(=O)(CCCCCl)Nc1c(C(=O)Nc2cc(C#N)sc2)scc1 55295,N#Cc1cnn(CC(=O)NCCCCCNC(c2cc(C3CC3)on2)=O)c1 55296,C(=O)(CCC(C(C)C)NC(=O)C(F)C(C)(F)F)NCC(CC)C(C)C 55297,N1(C(C2N(Cc3ccc(OC)cc3F)CC(O)C2)=O)C2COCC1CC(F)C2 55298,c1(C(=O)NCC2(O)CC(CNC(C(C)NC(N)=O)=O)C2)cn(C)c(=O)nc1O 55299,C1(NC(c2cncc(OC)n2)=O)CN(C(=O)C2=COCCC2)CC(F)(F)C1 55300,c1(OCC(=O)NCC2C3CN(C(c4cc(O)cs4)=O)CC23)cccc(F)n1 55301,CCCCC(=O)C(=O)NC(C)(CNC(=O)C=CS(C)=O)C1CCC1 55302,CCC(C(=O)N1CCCC1CCNC(=O)C=CI)C(C)C 55303,c1(C(c2nnnn2C)NCc2c(C)scc2)ccc(S(C)(=O)=O)cc1 55304,N1(C(C(C2CCCCC2)OC)=O)CCC(C2(O)CN(C(=O)C3=CSCS3)C2)CC1 55305,c1(C(CNC(=O)CCC2CC2(F)F)(F)F)ccc(Cl)cc1Cl 55306,c1(C(N2CCC(N(C)C(c3cc(C(C)(C)C)no3)=O)C2)=O)ccc(O)c(Cl)n1 55307,CC(C)CC(C)CC(=O)N1CCC(C(=O)NCCc2c[nH]nc2O)CC1C 55308,C1(CCOC)CN(C(c2cn(CCF)nn2)=O)CCN1C(=O)CN1CCOCC1 55309,c1(CC)cncc(C(=O)NC(C)CC2CCN(C(=O)C(C)(C)C3CCC3)CC2)c1 55310,N1(c2cc(OCC(C)C)ncn2)CC2CC(NC(=O)Cc3ccc(O)nc3)C2C1 55311,C1(C(=O)OC)C2CN(C(C3CCC4(CC4)C3)C(=O)NCCSC)CC12 55312,N1(C(CCC#CC)=O)CCCC(COC)(NC(=O)C=NOC)C1 55313,C1(NC(C2C(OC)CC2)=O)CCN(C(C2CC(SC)C2)=O)CC1(C)C 55314,C(C)(CNC(=O)C(C)OCC(C)C)(CC(C)C)NC(c1sc(CCC)c(CC)c1)=O 55315,N1(C(c2c(CCC)[nH]cc2)=O)CCC(C)N(C(c2c[nH]nc2C)=O)CC1 55316,c1(C(=O)NC2CC(C)(NC(C3C=CCC3)=O)C2)cccc([N+](=O)[O-])c1O 55317,N1(C(c2c(C)cc(C)o2)=O)CCC2(COC(CNC(c3cc(C)c(C)o3)=O)C2)C1 55318,c1(-c2ccc(NC(C3CCN(C)S3(=O)=O)=O)cc2)oc2ccccc2c1Br 55319,CC1CN(C(C2COCCN2C=O)=O)CCCN1C(=O)CCC(F)(F)F 55320,N1(C(C2CCCC2NC(=O)CC2CC3CCC2C3)=O)CCc2nncn2CC1 55321,C1(C2CN(C(=O)C(C)Oc3ccc(Br)cn3)C2)(OC(CC)(C)C)CC1 55322,c1(C(=O)NCCC(CNC(C2CC2(C)C)=O)OC)ccc(CO)cn1 55323,CC1C=C(C(=O)NCCCCCN(C)C(C2(C)CNC(=O)C2)=O)C1 55324,C1(C(N2C(CNC(C(CC)(C)CO)=O)C(C)CC2)=O)C2CCC1(C)C2(C)C 55325,c1(C(C)C)ccoc1C(=O)NC1CCN(CC2COCC2OCCC(F)F)C1 55326,C1(F)(C(=O)NC(C(C)C)CNC(=O)CCSc2nnnn2C)CC=CCC1 55327,Nc1nc2ncccc2cc1C(N1CC2(NC(C3CCC(=O)NC3)=O)CC1C2)=O 55328,C1(NC(CCNC(COC)=O)=O)CC2CCC(C1C)N2C(c1cccc(N)n1)=O 55329,Cc1ccc(C)c(C(N2CCC(N(C(=O)CN3CCP(C)(=O)CC3)CCO)C2)=O)c1 55330,c1(CN2CC(NC(c3c(C)cccc3)=O)(CO)C2)cccc2cccnc12 55331,c1(CNC2CCC(C(=O)Nc3c(C#N)cc(F)cc3)C2)ccc(Cl)c([N+](=O)[O-])c1 55332,S(=O)(=O)(c1ccc(NCc2ccncn2)c(Cl)c1)NC(c1cc(C)cc(C)c1)C 55333,Cc1cc(C(N2CCOC(C(C)Nc3ccncn3)C2)=O)c(C(F)(F)F)o1 55334,c1(OC)ccc(C2(CSC3CCC(NC(C4(OC)CC4)=O)C3)COC2)cc1Cl 55335,C1(NC(c2ccc(C(C)C)o2)=O)C=CCN(C(=O)CNC(=O)CCCCO)C1 55336,N1(CC(=O)NCC(CN(C)C(c2ccn(C)n2)=O)O)C(=O)NC(C)(C2CC2)C1=O 55337,Cc1cnc(C(N2CC(CF)(NC(=O)C(c3cncnc3)C)C2)=O)cc1Cl 55338,c1(OC)ccc(-c2cc(C(N3CCC(CC(=O)N4CCC4)C3)=O)c[nH]2)cc1 55339,CC(Cc1ccncc1)N=c1cc[nH]c(=NCCCc2ccccc2)[nH]1 55340,c1(CCC)nc(C(=O)NCCOCCCN(C(=O)C=CC(C)(C)SC)C)co1 55341,C(=O)(C1CCc2nccn21)NC1CN(C(C2(SC)CC2)=O)CC1C 55342,C1(C(=O)NC(C)CCNC(=O)Cc2cccnc2Br)CC2CCC1CC2 55343,c1(C(=O)NCCCN(CC(C2CCCC2)OC)C(C)C)cnc2ccccn12 55344,C=C1CCCN(C(=O)CSCCNC(c2ncn(CC)n2)=O)C1 55345,C(=O)(CCCCC(C)C)N1C(CNC(CCCc2onc(C)n2)=O)CC(C)(C)C1 55346,C(=O)(CC1CCc2ccccc21)NCC1CCC(NC(CSCC(=O)OC)=O)C1 55347,C12(C(=O)NC3C(C)N(C(c4ccc(CO)o4)=O)CC3)CC=CC(C1)OC2 55348,N1(C2CCC(NC(c3cc(C4CC4)on3)=O)C2)CCN(C(=O)C2=CCSC2)CC1 55349,Cc1ccc(CC(=O)NCCC(C)NC(=O)CC2CC(C3CC3)C2)cc1Cl 55350,c1(CCC(=O)NCC2(CNC(=O)C(C3CC3)C3CC3)CC2)ncc(F)cn1 55351,c1(C(N2CCCC(NC(CCC#CC)=O)C2)=O)cnc2cc(OC)ccn12 55352,Cc1ccn2cnc(C(=O)NC3C=CCN(C(C4CC4CC(C)(C)C)=O)C3)c2c1 55353,C1(CC(=O)NCCCOCCNC(C(C)c2cccs2)=O)CCOCC1(C)C 55354,C(=O)(C1CCc2cc(OC)ccc21)NC1CCC(NC(C2C(OCC)C2C)=O)C1 55355,C1(N(C(C2CCCN(C(C3C(C(C)C)C3)=O)C2)=O)C)CCCC(C)C1C 55356,C12(CNC(c3ncn(C)n3)=O)CCC(NC(C3CC4CC4C3)=O)(CO1)C2 55357,C=C=C(C)CC(=O)NCC1CC1CNC(=O)C(CC)c1cccnc1 55358,C1(C(C)(C)C)(C(=O)NCCOC2CN(C(CC3C(C)CCC3)=O)C2)CCCCC1 55359,c1(C(N(C(C)C(=O)NCCS(C)(=N)=O)CCC)=O)cc(C(C)C)no1 55360,c1(CNc2c(CC(=O)Nc3ncc(C)c(F)c3)cccc2)ccc(F)c(C)c1Cl 55361,c1(CC(=O)NCCC(CNC(C(C(C)O)C)=O)(C)C)ccc(S(N)(=O)=O)cc1 55362,c1(CC(=O)NC(CCNC(C(CC)NC(C)=O)=O)C)c[nH]c2cc(OC)ccc12 55363,c1(C(=O)NCC(C)N(C)C(c2cnn3c2NCCC3)=O)snc2ccccc12 55364,c1(OC2CCC2NC(CN(C(=O)OC)CN)=O)ccc(SC)cn1 55365,C1(C(NOCC2CC(=C)C2)=O)C2CC1N(C(=O)C=Cc1ccncc1)C2 55366,CCC1=C(C(=O)NC(C)(C)CCNC(=O)C(C)CC(F)(F)F)CCCO1 55367,c1(OC)cccc2ccc(CN3CCN(C4CCC(F)(F)CC4)CC3)nc12 55368,S(=O)(=O)(c1ccc(C(F)(F)F)cc1)N1CC2C(c3nnc(C(C)C)o3)(CC2)C1 55369,C(=O)(C(F)C(C)CC(C)(C)C)N(C)CC1CCCCN1C(=O)C(=O)N=S(C)(C)=O 55370,S(=O)(=O)(c1ccc(N2CCS(=O)(=O)CC2)c(Br)c1)NCc1ccc(OC)cc1C 55371,c1(CNC(C2CC(C)OCC2)=O)cnn2c1CN(C(C1CCN(C)CC1)=O)CC2 55372,C=CC1CN(C(=O)CCCn2ccnn2)CC1NC(=O)CC1CNC(=O)C1 55373,c1(N2CCN(C(=O)Cc3cc(F)ccc3F)C3C2C3)ncnc2cc(Br)ccc12 55374,Cc1nc(C)c(Cc2c(SC(N3CCC(c4cnn[nH]4)CC3)=O)nn[nH]2)s1 55375,Cc1cc(C)c(CN2CCN(C(=O)C=Cc3ccoc3)C3CC23)cc1C 55376,C=CC1(CC(=O)NCC2CN(C(c3cc(C4CCCC4)no3)=O)C2)CCC1 55377,c1(C(=O)Nc2c[nH]nc2C(=O)Nc2cc(F)ccc2I)cc2sccc2[nH]1 55378,c1(CC(=O)NC2(CO)CCN(C(=O)C3=CCC3)C2)cccc(F)c1 55379,C(=O)(C(CC)C(F)(F)F)N(CC)CC1CCCN1C(C1CS(=O)(=O)C1)=O 55380,C1(=O)C(C)(C)Cc2cn(nn2)CC(OC)CN1.c1(COC)cnc(SC)o1 55381,N1(C(CC=C)=O)CCC2CCC12CN(c1cn(Cc2ccccn2)nn1)CC1CC1 55382,N1(C(C2CC(=O)NC(=O)C2)=O)CCC2(CC1)CC2C(=O)Nc1ccc(O)cc1 55383,c1(CC)c(C(=O)N(CC(O)CN(C)C(c2ncccn2)C)C)cnn1C 55384,c1(C(C)NC(c2cc(C3CCC3)no2)C)coc2ccccc12 55385,c1(C(=O)NCCn2cc(CNC(C(C)C(F)(F)F)=O)nn2)cc2cccn2cn1 55386,c1(NCC2(CC)CCC2)nc(N2CC(OC)C(OC)C2)nc2sccc12 55387,CN1CCC(C)(C(=O)NCC2(C)CCN(C(C3(c4cc[nH]n4)CC3)=O)CC2)CC1 55388,C1(C(=O)NCC2CCC(NC(C(c3cnn(C)c3)C)=O)CC2)CC2CCC(C1)O2 55389,c1(C(=O)Nc2c(NC(COC3CC(C)(C)OC3)=O)cccc2)cc(O)ncc1F 55390,C(=O)(CS(=O)(=O)C(C)C)N1C(CNC(CC2(C=C)CCCCC2)=O)CC(F)C1 55391,CN1CCN(C(=O)Cc2csnn2)CC1CNC(=O)COc1ccon1 55392,N1(C(C(=O)NCCCC)CC2CCC(C(C)(C)C)CC2)CCC2C(O)C(C)(C)C12 55393,C(=O)(C#CC1CCCC1)NCCCCC(C)NC(C1(c2cccc(O)c2)CC1)=O 55394,C(=O)(C(C(C)CC1CC(F)(F)C1)N1CCCC(C(N)=O)C1)NCCCOC 55395,Cc1ccc(NC(C2C3CC3CN2C(=O)Cn2c(C)ccc2C)=O)cc1F 55396,c1(CC(=O)N(C2CCN(C(=O)C#CC3CCCO3)C2)CC)cccc2sccc12 55397,C1(NC(c2n(CCC)ccc2)=O)CCN(C(c2cn[nH]c2)=O)C1(C)C 55398,C#Cc1nc(C(N2CCN(C(=O)CCCCN3CCCCC3)CC2)=O)cs1 55399,N1(C(c2c(C)cno2)=O)CCC2(C1)CN(C(=O)CCc1nc(CN(C)C)no1)C2 55400,CC(=O)CCCC(C)C(=O)NC(CC(=O)N1CCCC(F)C1)CC(C)C 55401,CC1(C)COc2cc(C(=O)Nc3ncc(-c4cncc(F)c4)s3)nn2C1 55402,CCC(CC)C(C(=O)N1CC(C)(C(N2CC([N+](=O)[O-])C2)=O)C1)OC 55403,N1(C(c2ccc(C(C)C)o2)=O)CCCC(C)(CNC(c2cnc(O)c(Cl)c2)=O)C1 55404,Cc1cc(CN(c2nnnn2CC2CCSC2)C)cc(C)c1Br 55405,C#CC(C)(C)C(=O)NCCCC.c12nnc(n1CC(F)(F)F)CS2 55406,C1(C(=O)NCC(CC(=O)N(CCCO)CC)O)CC2C(C1)C2(C)C 55407,N1(C(CCC2CC(C)C2)=O)CCCC(CO)(CNC(=O)CS(C)(=O)=O)C1 55408,C(=O)(C(C)(C)CCCNC(C1CCC(=O)C1)=O)NCC(n1ccnn1)C 55409,C1(CC(=O)NC)CN(C(C2CCC2(C)C)=O)CCN1C(C1CCC=CCC1)=O 55410,C#CC(CNC(=O)C(Cn1cncn1)NC(=O)CN1CC(C)(C)C1)CC(C)(C)C 55411,n1(CC)nc(C2CC2)cc1C(N1CC(NC(=O)CCCc2cccs2)C1)=O 55412,C(=O)(C(O)P(C)(C)=O)N(CCCNC(=O)CCCc1cncs1)C 55413,c1(C(C)(C)C)ccc(CNc2ncccc2Br)cc1 55414,N1(C(=O)NCC(N2CCCCCC2)C)C2CCCC1CN(C)C2 55415,CC(C)CC(CCO)N=c1[nH]c2c(c(=NCC3(CO)CC34CCC4)[nH]1)COCC2 55416,C1(C(N2CC(C(C)(C)O)(CNC(C3C(C(=O)OC)C3)=O)C2)=O)CC2(C1)CC(F)C2 55417,Cc1c(NCCNC(=O)C(C)C)nc[nH]c1=NCc1ccc(NC(N)=O)cc1 55418,c1(C(N(C(C)C)Cc2cccc(C)c2C)=O)ccc2c(c1)OC(C)C2 55419,Cc1nccc(C(=O)NCC2(C)CCCN2C(=O)Cc2ccc(F)cc2Cl)c1O 55420,C12(C(=O)NCC(c3ccc(O)cc3)N(C(=O)C(Cl)=CCl)C)CC3CC1C2C3 55421,CC12CCCN1C(=O)c1c(cccc1)C(=O)NC2.c1(NC(N)=O)cnccc1Br 55422,C#CCC(CC#C)C(=O)NCCCC(CCC)NC(c1csc2c1CCCC2)=O 55423,C1(NC(CC(=O)OC(C)(C)C)=O)CC=C(C(=O)NCc2occ3c2CCC3)C1 55424,CC#CCCC(=O)N(CCNC(c1cncnc1-c1ccccc1)=O)C1CC1 55425,c1(SC)cncc(C(=O)NC2CC(NC(=O)C=CC3CCOC3)C2)c1 55426,N1(C(C2(CO)CCC(C)(C)CC2)=O)CCC(C2CCN(C(=O)C=CCO)C2)C1 55427,C1(NC(=O)CCN(C(c2scnc2Cl)=O)CC2CC2)CN2CCC1CC2 55428,N1(C(CCC=CCC=C)=O)CCC(C)(NC(=O)C(C)CC2CCC2)C1 55429,n1(CC(=O)Nc2c(C)cc(NC(=O)CSCC(N)=O)cc2)cnc2c1CCCC2 55430,C(C)(CCCC(=O)N(CC(C)CO)C)NC(C12CCC(OC)C1C2)=O 55431,C1(C(=O)NC(CCC2N(C(COC)=O)CCCC2)(C)C)(CF)CC2(CCC2)C1 55432,c1(NC(C(C(C)C)NC(C(CCC)NC(N)=O)=O)=O)cc(C#N)ccc1O 55433,N1(C(c2c(C)ocn2)=O)CCN(C(c2csc(CC(F)(F)F)n2)=O)CC1 55434,S(=O)(=O)(c1cccc(=NC2CCC=CCCC2)[nH]1)NC1CN(C)C2(C1)CCOCC2 55435,c1(N2CCC(N(C(=O)C(O)CCSC)CCC)C2)cc(C)c(C#N)cn1 55436,CC1CC(C(N2CCC(C(C)NC(C3(C4CC4)CCC3)=O)C2)=O)CCC1C 55437,c1(C(N2CCC(C3N(C(C(F)OC)=O)CCC3)C2)=O)ccc(F)nc1F 55438,C1(C(C)NC(C(C)=C(C)C)=O)CCN(C(c2cc[nH]c2C2CC2)=O)C1 55439,CC(CC(=O)c1cccc(Br)c1)C(=O)NCC(O)(Cc1ccccc1)C1CC1 55440,C1(NC(c2scc(OC)c2)=O)CS(=O)(=O)CC1NC(=O)C=CSC 55441,C(C)(C(=O)NC1CC(NC(c2cc(C)sc2C)=O)C(O)C1)(C(C)C)OC 55442,N1(C(C(C)OCCCC)=O)CC2(CCC(NC(C3C=C(C)CS3)=O)CC2)C1 55443,S(=O)(=O)(C=Cc1ccccc1)N1CCN(C(=O)C=Cc2ccccc2)C2C1C2 55444,n1(CC=C)ncc2c(O)nc(=NCC(C)CNC(=O)C(C)CC(C)(C)C)[nH]c12 55445,C(=O)(NN1CCCC1C(=O)NC1CCC2CC12)c1cc(C(N)=O)[nH]c1 55446,N1(C(C(C)NC(=O)NC)=O)CCCC(CO)(NC(=O)CC2C=CS(=O)(=O)C2)C1 55447,C1(N(C(C2C(CC)C2)=O)C)C=CC(CC(=O)N(C2CCCCC2)C)C1 55448,C1(NC(C2C(NC(CCCC3C(C)C3)=O)CCC2)=O)CCOC1(C)C 55449,C1(C(=O)NCCC2(CNC(=O)COC3CC(F)(F)C3)CC2)CCCCCS1(=O)=O 55450,c1(C(=O)NCCN(C(=O)CC2OCCCO2)CCC)coc(OC)n1 55451,C1(C(=O)NC(C)C(=O)O)CC=CC(n2cc(-c3ccc(F)cc3)nn2)C1 55452,c1(C(=O)NC(C(C)(C)C)CNC(C23CCC2CC3)=O)cc2n(n1)CCCC2=O 55453,C1(CN(C(=O)C(=O)N(C)C)C)CCN(C(C2CC(=C3CC3)C2)=O)C1.C1CN1 55454,C12(NC(COCC#C)=O)CCCC1CN(C(c1cc(CC)nnc1C)=O)C2 55455,CCC(c1ccnc(Cl)n1)=Cc1ccc(NC(c2ccn(C)c2)C)cc1 55456,N1(C(C(C)(C)OCC)=O)CCOCC(CNC(c2nc(C)n(C)n2)=O)C1 55457,C=CC1(C(N2CSCC2C(=O)NC(C)CC(C)C(F)F)=O)CCCCC1 55458,N#CC1CN(C(C2CCOC2)=O)CCN1C(c1ccc(N2CCC2)cc1)=O 55459,N1(C(=O)C=Cc2cccc(Cl)c2)CCCC2(CCC(NC(C3(F)CC3)=O)C2)C1 55460,c1(CC(C(=O)NC(C(=O)OC(C)C)Cc2ccccc2)N)cccnc1F 55461,c1(NC2CN(C(c3c(C)cco3)=O)CC23CCC3)c(Cl)cc([N+](=O)[O-])cc1Cl 55462,C(=O)(CC(C(F)F)NC(c1ncc[nH]1)=O)Nc1cccc(C(C)C)c1 55463,c1(NC(N2CCC(CC)C2)=O)cncc(OC)n1 55464,C1(CC)C(NC(C2CCC(CC)CC2)=O)CCCN1C(=O)CCn1ccnn1 55465,n1(CC(=O)N(C)CC2CCN(C(C3(COC)CCCC3)=O)C2)ncn(C)c1=O 55466,N1(C(c2c(NC(CC)=O)cccc2)=O)CC(C2CCCCC2)CC1C(=O)O 55467,N1(C(CCC=C)=O)CCC(C(=O)NCC2(c3ccnc(Cl)c3)CC2)CC1 55468,Cc1ccc2c(c1)CCC(C(=O)NCC1CCCCC1NC(c1csnn1)=O)O2 55469,C(=O)(C#CC1CCOCC1)NCCCC(CCC)NC(C1CCCC12CC2)=O 55470,N1(C(CC=C)=O)CCC(F)CC1C(=O)NCCC(O)CO 55471,C(=O)(C(C)CC(C)C)N.C(C(=O)NCCOCCCF)N(CC)CC 55472,CCC(Cc1ccccc1)CC(=O)NC12CC1CN(C(=O)CC(C)(C)C#N)C2 55473,c1(COC)cccc(CC(=O)NC2CCC2CNC(c2cccc(CO)n2)=O)c1 55474,C1(CC)CN(C(c2cc(=O)n(C)o2)=O)CCN1C(C1CCCOCC1)=O 55475,c1(OC)ccc(CNC(=O)NNC(C)Cc2ccccn2)c(F)c1Br 55476,C1(CC(=O)NCC2CCN(C(C3(O)CCSC3)=O)CC2)CCS(=O)(=O)C1 55477,Cc1cc(C(N2CCC3(NC(=O)CCCc4ccccn4)CC3C2)=O)nnc1O 55478,C1(C(N(CC(C)NC(=O)CNC(N2CCCC2)=O)C)=O)COC(C)CO1 55479,OC1COC2(CCN(c3ncc(-c4nn[nH]n4)cc3Cl)CC2)C1O 55480,c1(C(=O)Nc2cc(C)c(NC(c3ccnnc3C)=O)cc2)ccn2cncc2c1 55481,C(CCC(=O)NC1CC(C)(NC(c2ncsc2Br)=O)C1)OCC=C 55482,O=C(C1=CCOC1)NCC(C1CC1)NC(C1CCSC1)=O 55483,CCCCCCC(CC)C(=O)N1CCCCC1Cn1cc(CNC(N)=O)nn1 55484,c1(NC(CC2N(C(C3(CC)CC3)=O)CCOC2)=O)cnccc1[N+](=O)[O-] 55485,C1(CN(C)C(=O)N(C(C)(C)C)C)CC1C1CC1 55486,c1(CC)nc(N2CC=CC(NC(=O)C(c3cccc(C)c3)O)C2)c(C#N)cc1C 55487,Nc1ccc(C(=O)NC2(CNC(=O)Nc3ccccc3)CCC2(C)C)c(O)c1 55488,c1(C(=O)NCC(CNC(C(COC)(F)F)=O)F)cccc2c1ncn2C 55489,C(=O)(NN1CCCC1C(=O)NC1CC2(CCCCC2)C1)C1CCC(=O)N1 55490,c1(OC)cc(C)c(C(=O)NC2CCCC2CNC(c2c(C)coc2C)=O)cn1 55491,c1(C(C)C)ccc(OC(C)C(N2CCC(OC(C3CC(C#N)C3)=O)CC2)=O)cc1 55492,C1(C)(CNC(CN(C2CCC2)C)=O)CCCN1C(c1ccc(C(F)(F)F)nn1)=O 55493,C1(n2cnnn2)(C(=O)NC2(C)CN(C(c3cc(C4CC4)no3)=O)C2)CCOCC1 55494,N1(C(c2c(OC(C)C)n[nH]c2)=O)CC(NC(C23CCCC2C3)=O)C2(CCC2)C1 55495,c1(C(=O)NCC(CC)NC(C2C(CCC)CCC2)=O)ccc(C)cc1O 55496,Cc1nccc(C(=O)NC2CC(C(=O)N(CCO)CCO)C23CCC3)c1C 55497,c1(NC(C(C(C)O)NC(=O)CN)=O)cnc(F)c(F)c1 55498,CC1(C(=O)NC2CC(CO)N(C(=O)C3=COCCC3)C2)CC(C2CC2)=NO1 55499,C1(CC)(NC(c2ccc(Cl)c(OC)c2)=O)CCCN(C(=O)CN2CCCC2C)C1 55500,c1(C(=O)NC(CN(C(=O)C=CCF)CC)C)cc2c(OC)cc(OC)cc2[nH]1 55501,CC1(C(=O)NC2(C3CCC3)CC2)CCN(C(=O)C=CCN2CCC2)CC1 55502,Cc1cc(C)c(C(=O)NC2(C)CN(C(C34COCC3C4)=O)C2)cc1C 55503,N1(C(COCC)=O)CCC12CN(Cc1[nH]c(C)c(C(=O)OC)c1C)C2 55504,CC(C)C(C(=O)NC1CCN(C(C2CCS2(=O)=O)=O)C1C)Sc1ccccc1Cl 55505,c1(C(=O)NCC2N(C(C(C=C)O)=O)CCN(C)C2)ccc2[nH]ccc2c1F 55506,c1(NC(C)=O)ccc(C(=O)NCC2(O)CC(NC(C3CCC3(F)F)=O)C2)s1 55507,c1(C(=O)NC(CC2OCC(C(=O)OC)C2)=O)ccnnc1S 55508,Cc1cc(C(N2CCCC(N(C(=O)C(C)C3=CCCC3)C)C2)=O)cc2nc[nH]c12 55509,c1(C(=O)NC2C(CC)N(C(C)=O)CCC2)c(Cl)ccc(O)c1Cl 55510,Cc1[nH]c2ncccc2c1C(=O)NC(C)CCCNC(=O)CCC1CC1(F)F 55511,C(=O)(C1=CCCCC1)NC(C1CCN(C(c2ccc(SC(F)F)cc2)=O)C1)C 55512,C(=O)(C1=CC=CN2CCS(=O)(=O)N=C12)NCC(C)(CO)NC(=O)CCC(N)=O 55513,N1(CCN(C(=O)CC2CC=CCN2C)C)CCN(C(c2ccns2)=O)CC1 55514,C1(NC(CCc2ccc(CC)cc2)=O)CCC(C)N(C(C2C=CCCC2)=O)C1 55515,C(=O)(CC(C)n1ccc(C)n1)NCCN(C(=O)C=Cc1nnc[nH]1)CC 55516,CCCCCC(CCCCC)C(=O)NC1CC(NC(c2cc(C#N)oc2C)=O)C1 55517,Cc1cc(Br)c(N)cc1C(=O)NCCN(C(=O)CCCC(F)(F)F)C 55518,c1(C(=O)NC(CCNC(c2cn(C)[nH]c2=N)=O)(C)C)cccc2nsnc12 55519,N1(C(C2CC(C(=O)OC)C2)=O)CCC2(CC1)CC(NC(C1C3COCC13)=O)C2 55520,c1(C(=O)NC2(C)CC(NC(=O)CC3(C(F)F)CC3)C2)ccc2c(c1)C(=O)C(=O)N2 55521,C1(=CC(=O)NCC2CC2NC(=O)CCc2cc(Cl)cs2)CN2CCC1CC2 55522,c1(C(=O)NCC(C2N(C(C(C)C)=O)CCCC2)(C)C)cnn2c(=O)cc[nH]c12 55523,N1(C(c2cc(C)[nH]c2)=O)CCN(C(=O)CC(C)C(F)(F)F)CCC1C 55524,c1(C(=O)NCC(CNC(c2ncc(C)cn2)=O)O)c(N)sc2ccccc12 55525,c1(C(N2C3CC(CC(NC(CSCCC)=O)C3)C2)=O)ccc2n[nH]cc2c1Cl 55526,c1(NC(CC)C(=O)N(C)CC2(NC(=O)C(N)=O)CC2)cccnc1Cl 55527,C(=O)(C1=CCN(C(c2cnnc(O)c2)=O)C1)NC(C(C)C)CO 55528,N#Cc1ccc(C(=O)NC2CCCN(C(=O)C(O)Cc3ccccc3)C2)c(O)c1 55529,Cn1cc(C(=O)NC2CCCCC2CNC(=O)C(C)(C)c2cscn2)n(C)c1=O 55530,c1(CC(=O)NC2(COC)CCN(C(C3(C)CC(C)(C)C3)=O)C2)ccc(C#N)cc1 55531,C1(C(N(CC(C(=O)OC)C)C)=O)CC(C)(C)CN1C(c1cc(C)c(F)cn1)=O 55532,N1(C(CCOCC#C)=O)CCC(C)C(N(C(=O)Cc2csc(C)n2)CC)C1C 55533,CC(C)CC(C(=O)NCC1(C)CN(C(=O)C(C2CCOCC2)O)CC1C)N(C)C 55534,C(=O)(C1=CC2CCCCCC12)NC1(CO)CN(C(CN(C(=O)OC)C)=O)C1 55535,N(C(=NCCCSC)NCC1(OC)CCSC1)Cc1ccc(OC)cc1Br 55536,C(=O)(C(CC(C)C)n1ccnc1)NC(CC=C)CNC(C1(CN(C)C)CC1)=O 55537,c1(C(=O)NC2CCC(CNC(C3(C)CC4CCC3O4)=O)C2)ccc(Cl)c(N)c1Cl 55538,c1(C(N(C2CCCCN(C(=O)C(C)(C)CF)C2)C)=O)cn2ccc(F)cc2n1 55539,CCCCC(CNC(=O)CCCN(C)C(=O)OC)NC(C1CC(CC)C1)=O 55540,C1(OC)CC1C1CCN(C(C2(C#N)CCN(C(=O)OC(C)(C)C)CC2)=O)CC1 55541,Cc1nc(C(N2CCOC(C(C)NC(=O)C(C)C3CCCO3)C2)=O)[nH]c1C 55542,C1(CCC)(C)CCN(C(=O)C=CC(C)NC(=O)C(C)C2CCC2)C1.OC 55543,c1(C(=O)NCC2N(C(c3c(C)coc3)=O)CCC2)ccc([N+](=O)[O-])cc1Br 55544,c1(C(=O)NCCCC(C)NC(c2ccc(C)s2)=O)ccnc2c1CCO2 55545,Cc1ccc(C)c(OCCCNC(c2ccc(N)cc2Br)=O)c1 55546,Cc1onc(Br)c1C(N1CC(NC(=O)COCc2ccccn2)C(F)C1)=O 55547,c1(C(N)=O)cccc(NCC(=O)NCC2CC2NC(=O)Cn2cccn2)c1 55548,c1(C(N2CC(CC(=O)N(CCF)CC)OCC2)=O)ccn2ccnc2c1 55549,Cc1cc(C(=O)NCC2CC(NC(c3cc(Cl)sc3Cl)=O)C(O)C2)cn(C)c1=O 55550,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1C(CNC(CN(CC(C)(C)C)C)=O)C1 55551,C1(NC(=O)CSCC2CCCCO2)CC2(CCCN(C(c3cccnn3)=O)C2)C1 55552,N1(C(CC2ON=C(C)C2)=O)C(C(=O)N(C(CO)C(C)C)C)CC2CC12 55553,C(=O)(C(CO)C(C)(C)C)NCCCN(C(c1ccc(CC(C)C)s1)=O)CC 55554,S(=O)(=O)(C(F)(F)F)N1CC(c2ccccc2)(NC(c2cc(C(F)(F)F)c[nH]2)=O)C1 55555,c1(NS(c2n(C)c(Br)cn2)(=O)=O)nc2c(c(=NCCS(C)=O)[nH]1)CSC2 55556,c1(CCC=C)ccc(C(=O)N(CCNC(C2(c3ccc(F)cn3)CC2)=O)CC)cc1 55557,N1(CC(=O)Nc2ccc(C=C)cc2)C2CCC1CC(CO)C2.C(=O)(C(F)(F)F)NCC 55558,C12(C(=O)OC)CCC(CC1)N(C(c1cc(-c3ccccc3)co1)=O)C2 55559,C1(C(=O)NC2CCC(NC(c3cn(C4CC4)nn3)=O)CC2)OCC2CCCC1C2 55560,C1(CC(=O)NC(C(=O)OC)(C)C)CC(C)NC(=S)N1.c1(C(N2C(=O)C2)=O)cccs1 55561,c1(OC)cc(C)cc(-c2cccnc2C(N2CCCCC2C(N)=O)=O)c1F 55562,c1(CCC(=O)NCC2(F)CCC(NC(C(C)(C)C)=O)C2)c(F)cccc1F 55563,CC1(C)CC(NC(C2CC2)C2CC2)CC(C)(C)C1.C(=O)(CCCC1CC1)O 55564,Cc1cc(C(=O)NC(C(=O)N2CC(C(F)(F)F)C2)C2CCOC2)nn1C 55565,Cc1ncc2c(n1)CN(C(=O)OC(C)(C)C)C2C(=O)Nc1cnccn1 55566,N1(C(c2c(COC)cccn2)=O)CCC(CNC(=O)CCCN(C)C(C)C)C(O)C1 55567,C12(C(=O)NC(C3CCN(C(c4cc(F)ccc4F)=O)C3)C)CCCCN1CCC2 55568,CC1CC(NC(C2(C)CC2(F)F)=O)CCN1C(c1coc(O)n1)=O 55569,C1(C(=O)NCc2ccc(C#N)cn2)CN(C(=O)CCCC2CC2)CC12CCC2 55570,N12CC3(CCC1C3)C(=O)NCCNC2=O.c1(C(=O)N)cscn1.CC(C)(C)O 55571,C(=O)(C1CC=Cc2ccccc21)N1CC(NC(COC(C)(C)C(F)(F)F)=O)C1 55572,C(=O)(CCCC(C)(C)C#N)NCC(CNC(C(C(=O)OCC)C1CC1)=O)O 55573,c1(C(=O)NC2CCN(C(c3c[nH]cc3C3CC3)=O)CC2O)cc2ncccn2n1 55574,CCCC(C(F)(F)F)NC(=O)CSCCNC(=O)Cc1ccoc1C 55575,CN1CCN(C(=O)NC2CCC(N3CCOCC3)C2)CC1CC1CC1 55576,n1(CCNC(C(C2CC2)SC)=O)ccc(C(N2CC(c3nncn3C)C2)=O)c1 55577,N1(C(c2ccc(NC)cc2)=O)CCC(NC(=O)C=Cc2ccccc2)C12CC2 55578,C(CCC(=O)N1CCCC1CC(N1CC(N(C)C)C1)=O)N(C(C)=O)C 55579,C1(C(=O)OC(C)(C)C)CC(NCC(=O)N(CCCCC)CC(=O)OCC)C(O)C1 55580,N1(C(C=C(C)C)=O)CC(NC(C2CCOC2c2cccnc2)=O)CCC(O)C1 55581,C(c1ccc(O)c(OC)c1)=CC(=O)NC(CC)CNC(c1csc(C(C)C)n1)=O 55582,C(=O)(CCCNC(=O)OC)NCCCNC(C(C1CCC1)OCC)=O 55583,CC(CNC(c1cc(C(O)C2CC2)ccn1)=O)CC(=O)N(C(C)C(C)C)C 55584,CCCC(CNC(C1CCN(OC)CC1)=O)C(=O)NCCN1CC(C)(O)C1 55585,C1(C)(C(N(CCC)CCO)=O)CCN1C(=O)C(C1(O)CCCC1)F 55586,c1(SCCCC)nc(-c2ccc(N(C)C)cn2)nn1CCC(=O)NC(C)(C)C 55587,C1(C)(NC(C2C(CC)C2)=O)CCN(c2ccnc(-c3cc(OCCO)ccn3)n2)C1 55588,C12(C(=O)NCCN(C(Cc3cc(OC)no3)=O)C3CC3)CC(C)(CO1)C2 55589,c1(CCC(=O)NCC(C)NC(=O)C(C)OC2CCCCCC2)nnc(O)nc1O 55590,C(C)(C(=O)N1CCN(C(=O)COc2ccc(C)cc2F)CC1)(C(F)(F)F)OC 55591,N1(C(CCC2(C)CN(C(c3cc[n+]([O-])cc3)=O)C2)=O)CCC(C)(O)C(O)C1 55592,C1(C(=O)NC2CCC2O)CC12CCN(C(=O)Cc1cn[nH]c1)CC2 55593,CCC(C)(CC)C(=O)N(CCCCNC(=O)CNC(c1ccccn1)=O)C 55594,c1(C(N(CC(CN(C(c2c(C)cncc2)=O)C)O)C)=O)c(Cl)cccc1[N+](=O)[O-] 55595,c1(C(=O)NC(CCNC(c2c(C)nc(C)[nH]2)=O)(C)C)cccc2oc(C)cc12 55596,c1(C(=O)NC2CC(C)(CNC(c3n(CC)ccn3)=O)C2)ccc(F)cc1C 55597,c1(C(=O)NCC2C3CC2N(C(=O)C(O)C(F)(F)F)C3)cc2c(F)c(F)ccc2[nH]1 55598,c1(CNC(=O)CCc2cnc[nH]2)cc2ccccc2[nH]1 55599,C1(NC(C2N(C)CCOC2)=O)CC2CCC(C1)N2C(c1ccsc1S(C)(=O)=O)=O 55600,C1(NC(C(C)OC)=O)CCCCCC1CNC(=O)CC1(O)CCC1 55601,C(N=c1[nH]cnc(NCCC2COCCO2)c1C)c1cc(CC)c(F)cc1 55602,C(=O)(C1=NNC(=O)CC1)N1CCC(F)(CNC(c2c(CCC)occ2)=O)C1 55603,c1(C(=O)NC2C(NC(=O)C=CI)CC2)ccc(Cl)s1 55604,N1(C(C(C(=O)OC)OC)=O)CCCN(C(=O)C(C)CC(F)F)CC1 55605,CCC(O)C(C)C(=O)N1CC(C(=O)NCCNC(=O)C2=C(C)OCC2)C1 55606,c1(CN2C(C)(C(N(CC)Cc3ccccn3)=O)CC2)cccc(C(F)(F)F)c1Cl 55607,C(=O)(C1=CC2(CN(C(C3(C)CC(=O)N(C)C3)=O)C2)OC1)NCCCOC(C)C 55608,N1(NCCS(CC)(=O)=O)CCNC(=O)CC1C.C12=CC=C(C=C1)C2=O 55609,CC1(C)CN(C(=O)C(O)Cc2ccccn2)CCC1NC(c1coc(C#N)c1)=O 55610,CC1(C)CCOC1C(=O)NC1C=CCN(C(c2cnc(-c3ccccc3)s2)=O)C1 55611,CC(C)C(=O)C(=O)Nc1ccc(C2CCOCC2)cc1.C12CCCN(C1)C2=O 55612,N1(C(c2cc(COC)oc2C)=O)CC2CC(NC(=O)C3=CCCC3C)C1C2 55613,C1(NC(c2ccco2)=O)CCCCN1S(=O)(=O)N1CC(C#N)C1 55614,N1(C(c2ccccc2)C2(NCC)CC2)CC(O)C(N)C1 55615,C(CS(=O)(=O)CC(=O)NCC1(C)CN(C(c2ccc(O)cn2)=O)C(C)(C)C1)OC 55616,C(=O)(C(C)(C)C(F)(F)F)N(CCCCCNC(c1c(C)cn(C)c1)=O)C 55617,C1(C(=O)NC(CCOC)C(N2CC3(CCOC3)C2)=O)CC2(CCC2=O)C1 55618,O=C(CCCCCNC(c1ncncc1Br)=O)Nc1ccccc1 55619,C1(C)(CNC(c2ccc(OC)cn2)=O)CN(C(=O)CC2(CO)CC2)C(C)(C)C1 55620,C(CCF)(C(=O)NCC1CC1(Cl)Cl)NC(Cc1cn(CC)nn1)=O 55621,C(=O)(C#CC(C)(C)CNC(=O)CC1CCC(O)C1)N1C2CC(OC)C2CC1 55622,CC(C)C(F)C(=O)NCC1(CNC(=O)CCc2ccc(Br)cc2)CC1 55623,Nc1ccnc(C(N2CC3(CCC3NC(c3csc(CO)n3)=O)C2)=O)c1Cl 55624,c1(C(=O)NC2CC(NC(C(C)N(C)C)=O)C(O)C2)cc(F)cc(S(N)(=O)=O)c1 55625,c1(C(=O)NC(CNC(C2(NC(N)=O)CC2)=O)CO)cc2n(n1)CC(F)C2 55626,c1(CC)ncc(C(=O)N(C(CNC(c2ccnnc2O)=O)CC)C)cn1 55627,CC(C)CC(C)(CNC(=O)CC1CC1)NC(c1ccc(N2CC=CC2)cc1)=O 55628,C#CCCCC(=O)NCCOCC(N1CCCC1C1CCCC1)=O 55629,C1(CNC(C2N(C(C)=O)CCC2)=O)CC2(CO1)CN(C(c1sccc1C)=O)C2 55630,C12(C(=O)NCC(CC=C)NC(C3CC4C=CC3O4)=O)CCC(O)(CC1)CC2 55631,CC(C)CC(C(=O)N1CC(NC(C2(C)CCN(C)C2=O)=O)CC(F)C1)C(N)=O 55632,Cn1c(C(=O)NC2COCC2NC(c2scnc2C(C)(C)C)=O)cc2ccsc12 55633,N1(C(c2c(C)ocn2)=O)CCC(NC(=O)Cn2cc(CO)nn2)C12CC2 55634,c1(N(C)C)cccc(C(N2CCC2CNC(C2CCN(C)C2=O)=O)=O)n1 55635,N1(C(CC(=C)C)=O)C2CCC1C(F)C(NC(c1nc(Cl)ccc1Cl)=O)C2 55636,C=CCC(C(=O)NCC1CC1CNC(C1CC2(CC2)CO1)=O)C(C)C 55637,c1(OCC(=O)NCCC(C)(C)NC(C(COCC)C)=O)cccc(F)c1F 55638,O=S(=O)(c1cnccc1N1CCCC(c2nncs2)C1)NCc1ccccc1 55639,C(N=c1cc(C)[nH]c(=NCCC2CCCC2(F)F)[nH]1)c1c(OC)ccnc1O 55640,CC1(CC(=O)NCCCNCCCNC(=O)CCc2cscn2)CCCC1 55641,C1(O)(CC(N2C(CC(C)C)CCC2)=O)CCN(C(C2CCCC2)=O)CC1 55642,CC(C)(C)C(CNC(c1ccc(=N)[nH]c1)=O)C(=O)NC1CC2CCC1O2 55643,CCCC(O)C(=O)NC1CC(F)(CNC(=O)CC2CCN(C)C2)C1 55644,C(=O)(C(F)(F)CCn1cc(CCC(=O)N(C)C)nn1)NCCC(C)N1CCCC1 55645,c1(C(N2CCC(OCCNC(C=COCC)=O)C2)=O)cnn2cccc(Br)c12 55646,Cc1cc(CC(=O)NC2CN(C(c3cccnc3C)=O)CC2C)cc(O)n1 55647,C1(NC(C2CCC(C)O2)=O)CC1C1CCCN(C(C2(CO)CC2)=O)C1 55648,c1(CCCC(N2CC(O)(CCNC(CC(C)O)=O)C2)=O)ccc(CN(C)C)cc1 55649,N1(C(C2(CC)CC2(F)F)=O)CCCN(C(=O)CC2CNC(=O)C2)CC1 55650,N1(C(C2(C)CCCOC2)=O)CCN(C(c2cc(CO)on2)=O)C(CCO)C1 55651,CC(c1cccnc1)=CC(=O)NC1(C)CCCN(C(=O)CC2C=CS(=O)(=O)C2)C1 55652,Cc1ccc(OCC(=O)NCCCC(C)NC(C2(S(C)(=O)=O)CC2)=O)cc1 55653,C1(C(N2CCC(C(C)NC(C3CCSC(C)C3)=O)C2)=O)Cc2ccccc2N1 55654,c1(C(=O)NCC2C(NC(C(CC=CC)C)=O)COC2)coc2cc(F)ccc12 55655,C(=O)(CC1CCOc2ccccc21)NC(c1ncccc1C)C(=O)OC 55656,C(N=c1nc(N2CCC(N3CCOC3=O)C2)c2ccc(C)cc2[nH]1)C1C=C(C)CC1 55657,c1(N(CCOCCN(C(C(CC(=C)C)NC(C)=O)=O)C)C)cnn2ncccc12 55658,C1(C(=O)NC2C(NC(C34CC(C(C)(C)C)(C3)C4)=O)COC2)COC(=O)N1C 55659,N1(C(=O)Nc2c(OC)cc(C(N)=O)cc2)CC2(CCCC2)C1c1ccco1 55660,c1(OC(C)(C)C)ccc(C(N2CCC2CNC(C23C=CC(CC2)C3)=O)=O)cn1 55661,Cc1cc(Cl)c(Cl)cc1C(N1CC2CC2(C(=O)Nc2ccnc(O)c2)C1)=O 55662,C1(C(=O)NCC2(C)CC2)CC2(CCN(C(=O)Cc3cccs3)CC2)C1 55663,CC(C)(C)C(=O)CCC(=O)N1CC(C(=O)NC2CC(=O)N(O)C2)C(C)(C)C1 55664,CC1ON=C(C(=O)NCCOC2CCN(C(c3cc(O)nc(O)c3)=O)C2)C1C 55665,c1(C(N2CCC(F)(n3cc(C4(C)N(C)CCC4)nn3)C2)=O)cnc(N)c(N)c1 55666,C=CC1(CC(=O)N(CC(C)O)CCNC(=O)C(C)CC2CCC2)CCOCC1 55667,C(c1ccccc1)=C(C(=O)NC(COC)CNC(C1(CO)CCCC1)=O)C 55668,C(=O)(CS(=O)(=O)CCO)NCC1C(CNC(C=Cc2c(C)cccn2)=O)C1 55669,Cc1nc(=N)[nH]c(=NCC(C)NC(c2ccc(F)o2)=O)[nH]1 55670,C(=O)(CC(C)(C)CC(F)F)N(C1CCCC1)C(C1(O)CNC1)C 55671,c1(OC)ncc(CNC2CCC(C(=O)Nc3cnc(C)nc3)C2)cn1 55672,c1(CC)cccc(C(=O)NC2CC23CC(NC(=O)CCNC(=O)CC(C)C)C3)c1 55673,C1(OCC#C)CCCN(C(C2CCC=CC2NC(=O)CC2CCOC2)=O)C1 55674,c1(CC(=O)NC2CCN(C(=O)C(F)CC3CCC3)C2)ccn(C(CC)CC)n1 55675,CC(C)CC(C(=O)NC1CN(C(c2cnn(C)c2C#N)=O)CC1O)NC(N)=O 55676,CC1(C)CN(C(c2ncoc2CN)=O)CC(CNC(=O)CCC2(C)CC2)O1 55677,Cc1nc2cc(C(=O)NCC#CCNC(=O)CC3CC(O)C34CCC4)ccc2o1 55678,c1(C(=O)OCC)ccc(C2CCCCN2C(C2COC(C)C2)=O)n1C 55679,C(=O)(C1(C)CCc2ccccc21)N1CC(F)CC(NC(COCC(=O)OC)=O)C1 55680,CC(O)C(C)(C)C(=O)N1CSCC1C(N1CC2CSCC2C1)=O 55681,C(=O)(C1CCc2nccn21)N1CC2N(C(c3cc(OC)cc(C)n3)=O)C(CC2)C1 55682,C(C(=O)NN1CCCC1C(=O)N(CC1CC1)CC1CC1)c1c(N)cncc1 55683,S(=O)(=O)(c1ccc(Cl)cc1F)NC1C(C#N)CN(C(=O)Cc2cccs2)C1 55684,c1(SCCNC2OCCN(C(c3ccccc3)C)CC2)c[nH]c2cc(F)ccc12 55685,C(CCc1ccccc1)(C(F)(F)F)NC(C(n1ccc(C2CC2)n1)C)=O 55686,Nc1cc(F)cnc1C(=O)NC1CC(CCNC(c2sccc2C2CC2)=O)C1 55687,N#Cc1ccsc1C(=O)NCc1ncccc1C(=O)NOCC1CCCCC1 55688,C=CC1CN(C(C2CCCC2NC(=O)CNc2ncccn2)=O)CCO1 55689,C(=O)(C(CC(C)(C)C#N)N1CCC(CCN2CCC2)CC1)NCCCSC 55690,C1(CCC)CN(C(=O)Cc2nccn2C)CC1NC(c1nscc1C)=O 55691,C(=O)(C1(C)CCn2ccnc21)NCC1(CNC(C=Cc2cn(C)nc2)=O)CC1 55692,c1(C(N(CCNC(CC=CCC)=O)CCC)=O)cc(Cl)cn1CC 55693,N1(C(C2(CC=C)CN(C(=O)CCSC)C2)=O)CCC2(CCC(OC)C2)C1 55694,C1(NC(CCCCCC)=O)CN(C(c2cnn(C(C)C)n2)=O)C2(CCOC2)C1 55695,C1(C(N2C(C(=O)NC3C(C(C)(C)C)C3)C(O)CC2)=O)CC2CC(=O)C1O2 55696,CC1(C)CC(NC(C2(CO)CC2)=O)CN1C(C1CCCCC1C(N)=O)=O 55697,C(=O)(C1c2c[nH]nc2CN1C(C1CC12CCCCC2)=O)NC1CC(CC(=O)OC)C1 55698,c1(OC)cc(F)c(C(N2CC(NC(C34CSCC3C4)=O)CC(F)(F)C2)=O)c(F)c1 55699,C=CCCCCC(=O)N(CC(C)N(C)C(C1CCN(CC)CC1)=O)C 55700,C1(C(=O)NCC(C(C)C)NC(C2CCN(C3CCCCC3)C2)=O)CCCC2CC12 55701,c1(C(=O)NCC2C(NC(C(CCSC)O)=O)C2)occ2c1CCOC2 55702,c1(C(=O)NC2C(NC(C=NOC)=O)COC2)cnc2c(c1)NC(=O)CS2 55703,N1(C(C2(C#N)CCCC2)=O)CCC2CCC(C1)N2C(C1CCCS(=O)(=O)N1)=O 55704,C(=O)(CC(C)C(F)(F)F)NCC(C(=O)N(C)Cc1nnc(C)o1)N(C)C 55705,c1(C(CO)NC(C2C(NC(=O)C=Cc3ccccc3)C2)=O)cc(F)ccc1F 55706,N1(C(C(N2CCSCC2)C)=O)CCCOC(CCNC(=O)CC(C)CN(C)C)C1 55707,C=CCCC(C)(C)C(=O)N1CC(CNC(=O)CC(C)N(C)C)C(O)C1 55708,C1(C)(NC(C=CCCC)=O)CCN(C(=O)Cc2c[nH]c(=N)nc2O)CC1 55709,C(=O)(C(O)C(C)(C)C)Nc1cc(C)sc1C.C12CC1NC(=O)C1C(C1)C(=O)N2 55710,c1(C(N2CC3(CCCN(C(C(C)C(F)F)=O)C3)C2)=O)cn(C)c(=O)c2cncn12 55711,c1(C(N2CCC(NC(C3C(CC(C)C)C3)=O)CC(O)C2)=O)ccc(F)c2occc12 55712,N1(C(c2c(OC)nsc2OC)=O)CCC(NC(c2ccon2)=O)CC1C1CC1 55713,CC1c2cc(Br)ccc2OC1C(=O)Nc1coc(C(C)(C)C)n1 55714,N1(C(C(C(=O)OCC)F)=O)CCN(C(c2cc(CC(C)C)on2)=O)C(COC)C1 55715,C(=O)(C1=C(C#N)CCC1)N(C(C)CC(=O)N1CCC(CCCO)C1)C 55716,C12(C(=O)NC3CC(C(C)C)OC3)CC(CN(C(c3cc(C#N)n(C)n3)=O)C1)C2 55717,C12(NC(c3ccc(OC)nn3)=O)CCC(CNC(=O)C(O)C3CCC3)(CC1)OC2 55718,C(=O)(C(=O)C(C)CC)N(CC(=O)NC(COCC)C)CC1CC1 55719,C(C)(C)(C(=O)NO)NC(CCNC(c1ccncc1)C)=O 55720,N1(C(CCC2OCC(C)(C)C2)=O)CCOCC(NC(c2cccc(Cl)c2Cl)=O)C1 55721,c1(CC(N2CCC(CCNC(CC(CC)OC)=O)CC2)=O)ccc(OC)cc1F 55722,C(C1=CCCSC1)(c1nnnn1C1COC1)Nc1cccc(C(N2CCCC2)=O)c1 55723,c1(C(N(C)CC2N(C(C3ON=C(CC)C3)=O)CCOC2)=O)ccc2ncnn2c1 55724,S(=O)(=O)(c1ccc(N2CCC(C)C2)cc1Cl)NCc1cccc(OC)n1 55725,C(=O)(CC(C)C(F)F)NCc1c(C(N2CCCC(C(=O)NC)C2)=O)nco1 55726,CC1c2c[nH]nc2CCC1C(=O)NC1CCN(C(=O)C(=O)C(C)(C)C)CC1C 55727,c1(C(N(CC(C)NC(C(C(C)C)OCC)=O)C)=O)ccc(Cl)cc1[N+](=O)[O-] 55728,C(CCC(C)C(=O)NCC1(CNC(C23CSCC2C3)=O)CC1)OC 55729,C(=O)(C1SCc2cccnc21)N1CC(CNC(COCCC)=O)C(F)(F)CC1 55730,c1(OCC(=O)NC2CN(C(=O)Cc3ccon3)C2)ccc2c(c1)CCCC2 55731,C(CC(C(=O)N(C)Cc1ccoc1)NC(c1c[nH]nc1C)=O)OCC 55732,N1(C(COc2cccc(C)c2)=O)CC(NC(=O)CC(C)F)CC(C)C1 55733,c1(OC)ccc(C(=O)NC2CCN(C(c3nc(C)nn3C)=O)CC2C)c(F)n1 55734,C(=O)(C#CC1CCCOC1)N(CC)CC1CCCN(C(=O)CCC(F)(F)F)C1 55735,C1(C(C)C)CN(C(c2cncc(F)c2)=O)CCN1C(C1CCC(C)O1)=O 55736,c1(OC)cc(CC(C(=O)O)NC(c2ccc(C(C)=O)o2)=O)ccc1O 55737,CCCCC(C(=O)N1CCN(C(C2OCCCO2)=O)C(COC)C1)C(C)C 55738,C(=O)(CCC(N)=O)NC(C(=O)NCCSC)CSC 55739,CC1OCCC1CC(=O)N(CCNC(c1ccc(C2CCOC2)s1)=O)C1CC1 55740,Cn1ncc2cc(CN3CC4CCN(S(=O)(=O)c5ccccn5)C4C3)ccc12 55741,N1(C(C2(C(F)(F)F)CCOCC2)=O)CC2CC(C1)C2N=c1[nH]ncs1 55742,N1(C(c2cnn(CC)c2Cl)=O)C2CCCC1CN(C(C13CCCN1CCC3)=O)C2 55743,N1(C(C(Cc2ccc(OC)cc2)C)=O)CCN(C(=O)CSC)C(C(F)F)C1 55744,c1(CC)c(C(=O)N(C)CC2CCN(C(=O)CNC=O)C2)nnn1C 55745,N1(C(c2cc(C(C)C)no2)=O)C(C(=O)NCCOC(F)(F)F)CC2CCCC12 55746,C(C(N=[N+]=[N-])C(=O)N1CC(NC(C2CC2(C)Br)=O)CCC1C)OCC 55747,CN1CCN(C(c2cc(Cl)cs2)=O)C(C(N2CCCC2(C)C2CCC2)=O)C1 55748,C(CC(=O)N=c1ccn(CCF)[nH]1)(C(F)(F)F)NC(C1(C(C)C)CC1)=O 55749,c1(NCc2ccccn2)ccc(-c2cncnc2)cc1 55750,Cc1ccc(C(=O)NCC2CCCCN2C(c2cncc(CO)c2)=O)c(N)n1 55751,c1(C(=O)NC(C2CCN(c3nccc(OC)n3)CC2)C)cc(F)cc(Br)c1C 55752,CCCC(CCC)=CC(=O)NCC1(CNC(C2CN(C3CCC3)C2)=O)CC1 55753,CC(C)C1=NOC(C(=O)N(C)CC2(O)CCCN(C(=O)C=CC(C)(C)SC)C2)C1 55754,Cc1ccnc(C(=O)NCC2CCCC(NC(=O)CNC(c3cscn3)=O)C2)n1 55755,C(=O)(C1=CC2C=CC(C1)C2)NC1CC2(C(NC(c3coc(Cl)n3)=O)C2)C1 55756,C1(NC(c2nc(-c3ccc(C)o3)sc2)=O)CN(C(C2(O)COC2)=O)CC1C(F)F 55757,c1(C(=O)NCCC(CNC(CCc2cc(C)on2)=O)O)cccc(CC#N)c1 55758,C(CCN=c1[nH]c2ccc(Br)cc2s1)OCCNC(C1CC2C=CC1C2)=O 55759,c1(C(=O)NC(C(C)NC(CC(CC)OC)=O)(C)C)ccc2nnn(C)c2n1 55760,CC1(CNC(c2ncoc2-c2cccs2)=O)CCCN1C(=O)CSS(C)(=O)=O 55761,C#Cc1cnc(C(=O)N(CCC(C)NC(c2cccc(CC)c2F)=O)C)c(C)c1 55762,n1(CC)c(SCC2CCCC(N)C2)nnc1-c1ccccc1 55763,c1(NCC(=O)NCc2ccc(N(C3CCCC3)CC)cc2)cccc(F)c1[N+](=O)[O-] 55764,C1(CC)(CC)CC(NC(=O)CN2CCOCC2)CN1C(=O)C#CC(=O)N(C)C 55765,c1(CNC(C(CNC(c2cc(CC)oc2C)=O)N(C)C)=O)nn(C)c(=O)n1C 55766,c1(C(=O)NC(C(=O)NCC(N2CCCC2)C)c2ccco2)cccc(O)c1F 55767,C1(OC)CCN(C(=O)CC2CCN(C(=O)C(N)=O)CC2)C1C 55768,C1(C(=O)NC2CC(NC(c3ccc(C)s3)=O)C23CCC3)Cc2nccnc2C1 55769,C(=O)(C(C)CCCOC)N1C(CC(NOCC(CC)C)=O)CCC1 55770,C1(CNC(CCOCC#C)=O)CC2(CO1)CN(C(=O)C(C)(C)CC=C)C2 55771,C1(CNC(c2cc(=N)[nH]cc2)=O)CCC2(CO1)CC(NC(=O)CNC(N)=O)C2 55772,C1(C(N(C)CC2CN(C(CC=CC)=O)C2)=O)CCC(C)C1 55773,C12(CNC(C3CC(C#C)(O)C3)=O)CCCC1N(C(=O)Cc1occc1C)CCC2 55774,c1(OCOC)ccc(C(=O)NC2CC2c2ccc(-n3cnnn3)cc2)cc1 55775,n1(CC(C)C)nc(CO)nc1-c1ccc(COc2cccc(C(C)(C)C)c2)nc1 55776,C(CCCC(C)NC(C1CC12CC2)=O)NC(C1(CCOC)CC1)=O 55777,C=C1CON(C(=O)CC2CCN(C(=O)COc3ccc(C)cc3)C2)C1 55778,N1(C(C(COC)(C)O)=O)CC(NC(c2ccc(OCCF)cc2F)=O)CC(O)C1 55779,N1(C(=O)NC(CC(C)C)c2ccccc2)CCc2cc(Cl)ccc2C1 55780,C=CCC(C)C(=O)NCCN(C1CCCC1)C(c1cnn(C)c1COC)=O 55781,C1(NC(C(c2cn(CC)nc2)=O)=O)CCCCC1CNC(c1coc(Cl)n1)=O 55782,N1(C(CCCOC)=O)CCN(C(=O)C(N2CCC(C)CC2)=O)CC1.C1(=O)CN1C 55783,C1(C(N(CC(C)O)CCNC(c2ccn(CC(F)F)n2)=O)=O)CC12CC(F)(F)C2 55784,C1(O)(C(C)NC(Cc2n(C(C)C)cnn2)=O)CCN(C(=O)C=CC2CCOC2)C1 55785,CC(CC(=O)N(C)CC1CCCCN1C(C1CCCO1)=O)P(C)(C)=O 55786,CC(C)C(CNC(C12CCC(CC1)C2)=O)C(=O)NC1CCCC(O)C1O 55787,CCCC(CCC)=CC(N1CCC(CNC(=O)Cc2nc[nH]n2)(OC)C1)=O 55788,CC(C)CC(O)CC(=O)NC(C1CCCN1C(=O)CCC1CC1(F)F)C 55789,C1(OC(C)(C)C)CCN(CCNC(C2(F)C(CC(=O)NC(C)(C)C)C2)=O)CC1 55790,C(=O)(CCCCCO)N1C(C)CC(NC(c2ccc(C(=O)CF)cc2)=O)C1 55791,N#Cc1c[nH]cnc1=NCC1CCCN(C(c2cccc3nc(O)oc23)=O)C1 55792,C1(CNC(C2(C(F)F)CC(=C)C2)=O)CC2CCC(C1)N2C(=O)CC(C)SC 55793,C1(C(=O)NC)CS(=O)(=O)CCO1.[N+](C)(C)(C)CCN 55794,c1(C(C(=O)NC2CCCC2)N(CCOC)C)cc(OC)c(F)cc1F 55795,N1(C(C(=CC2CCCC2)C)=O)CCCC(CCNC(c2cc(C)ccn2)=O)CC1 55796,c1(C(=O)NCC2N(C(c3c(C)cn(C)c3)=O)CCC2C)cc2c(C)n[nH]c2cn1 55797,C12(C(=O)NCC(CC)NC(c3cc(C(N)=O)n[nH]3)=O)CC(c3ccccc3)(C1)C2 55798,c1(CN2C(C(=O)Nc3ccc(CCO)cc3)CC(F)(F)C2)cc(Br)c(O)cc1O 55799,C#CCC(C)(C)C(=O)N1CCC(COC)(NC(C2CC2CC(C)C)=O)C1 55800,c1(CC(N2C(C)(CNC(C(C)OCCC#C)=O)CCC2)=O)cc(F)cc(Cl)c1 55801,c1(C(=O)NCC(CNC(CC2CC(=O)NCCC2)=O)O)ccc(F)c2ccsc12 55802,c1(NCC(C(C)C)O)ccc(S(=O)(=O)NC2CC3OCCCC23)c(Br)c1 55803,N1(C(C(CO)OC)=O)CCN(C(c2cc[nH]c(=N)c2)=O)CC1C1CCC1 55804,C(=O)(CC1CCCc2c1[nH]c1ccccc21)NC1C(C(=O)OC)C2CCC12 55805,C1(CNC(=O)C2=CCCCCC2)CN2CCCCC2CN1C(=O)Cc1ccon1 55806,C1(CC(N2CCCC(Cn3cc(CSCCO)nn3)C2)=O)C=CS(=O)(=O)C1 55807,N1(C(CCSC)=O)CCCC(O)(c2cn(Cc3ccc(=O)n(C)c3)nn2)CC1 55808,C1(OC)CC2CC(N(c3ccccc3)C(=O)CC3CCN(CC(C)C)C3)CC12 55809,N1(C(CCOCCOC)=O)CCC2CN(C(c3nccc4[nH]ccc34)=O)CC12 55810,C1(C(N2CC(CCC)C(NC(C3CCOC3(C)C)=O)C2)=O)COCC(C)(C)O1 55811,N1(C(COC(CC)C)=O)CCCCC1CN(C)C(c1sc(F)cc1Br)=O 55812,c1(NC(=O)CC(O)Cc2ccccc2)cccc2oncc12 55813,c12cc(cc(Cl)c1)SC2.C1(CCn2cc(CCN)nn2)CCS(=O)(=O)N1 55814,C1(OC)CN(C(=O)C(=O)NCCNC(=O)Cc2ccccc2)CC1CC(C)(C)C 55815,C1(NC(CC2(C)CC2(Cl)Cl)=O)CC2CC(C1)N(c1ncc(Br)c(O)n1)C2 55816,Cn1cncc1C(=O)NCc1ocnc1C(=O)NCCC1CC1C1CC1 55817,Cc1cc(-c2nc(Cc3ccc(F)cc3)nn2CC2CC2C)oc1Br 55818,C1(O)(CCNC(=O)C(O)C2CCC2)CN(C(=O)CC2CCOC2=O)C1 55819,C(C(CC(C)C)C(=O)N1CCOCC1CNC(c1cn2cnnc2cn1)=O)OC 55820,c1(C(=O)NCC(C)N(C(c2cccc(CC)c2)=O)CC)cnc2n1CCC(C)C2 55821,Cc1cnc(CCN2CCCC(C(N3CCCC(N(C)C)C3)=O)C2)cn1 55822,C(=O)(C1(C)OCCc2ccccc21)NCC(C(C)C)(C)NC(C12CC(CO1)C2)=O 55823,c1(C(=O)NC2(CN(C(C(CC)COC)=O)C)CC2)cc(S(N)(=O)=O)ccc1F 55824,c1(NC(C2CCC(C)(C)CC2)C(=O)OC)cc(=O)n2cc(Cl)ccc2n1 55825,c1(COC)ccc(OC23CC(CN4CCC(CN)C4)(C2)C3)c(C(=O)OC)c1 55826,c1(OCCOC)cncc(C(=O)NCC(O)CNC(=O)CC(C)(C)O)c1 55827,CCCCC(O)C(=O)NC(C1CCN(C(c2cccc(CN(C)C)c2)=O)C1)C 55828,C1(CNC(C2CC2C(F)(F)F)=O)COCCN(C(c2cnco2)=O)C1 55829,C(c1cccnc1)=C(C(N1C(CCNC(C(C=CC)O)=O)CCC1)=O)C 55830,c1(C(C(=O)NCCCSC)N(CCC=C)CC)nccc(Cl)c1F 55831,c1(C(C(=O)NC(C)C)N(CC=C)Cc2cccnc2)c(Cl)c(C)nn1C 55832,c1(CC(=O)N(c2cccnc2)CC=C)ccoc1C 55833,c1(C(=O)NCC2CN(C(=O)C(F)(F)CC3CC3)CC2(F)F)cccc2c1CCO2 55834,N1(C(C(c2ccccc2)C)=O)CCC(CCCNC(C2CC2Cl)=O)CC1 55835,C(=O)(C(C)C1=CCCC1)N1CCCCC(N(C(c2cccc(C#C)c2)=O)C)C1 55836,CC(C)CCN=C(NC1CN(C(=O)OC(C)(C)C)C1)NC1C(O)CC(O)C1O 55837,CCC(C)C(C)N(C(C1(CNC(=O)C(C)c2cc[nH]n2)CC1)=O)C1CC1 55838,CCC1=NOC(C(=O)NCC2CC(C)N(C(=O)CCc3cnccn3)C2)C1 55839,c12ccc(nc1)c(=O)[nH]2.CCC(C(=O)NCC(C)(O)C1(C)CC1)NC(C)=O 55840,c1(C(=O)NCC(=O)N(C(CNC(=O)CCNC(=O)C2CC2)C2CC2)C)cc[nH]n1 55841,C(CC(C)C(=O)NC1CC(CCNC(c2cnc(N3CCOCC3)s2)=O)C1)OC 55842,c1(N2C(=O)CC(C(N3CCC(OC)C3)=O)C2)ccc(Cl)c(F)c1 55843,c1(CC(N2CCC(C(C)NC(C3(CC=C)CCC3)=O)CC2)=O)ccc(F)c(C)c1 55844,CCCCCCC(C)C(=O)NC(CC1CCC1)C(N1CC2CCC(C1)C(=O)N2)=O 55845,CC(Cc1ccnn1C)C(=O)N1CCC1CNC(=O)CCc1ccccc1 55846,c1(N2CC(C)C(CO)CC2)nc2c(c(=NCCN(C)C)[nH]1)CCCCC2 55847,c1(CNC(C=C2CCC(C)CC2)=O)cc(O)nc(CNC(=O)CC2OCCO2)n1 55848,Cc1ccc2c(c1)C=C(C(=O)NC1CCOC(CNC(C3CC3F)=O)C1)CO2 55849,N1(C(C(CCC)O)=O)CC2CC(C1)CN(C(=O)C(F)C(F)(F)F)C2 55850,C(=O)(C(CC1CCCCC1)C(C)C)N1CCC(N(C(CCC)=O)C)CC1 55851,C(CC(F)CN=[N+]=[N-])NC(C(CC=CC)NC(C1OC2CCC1C2)=O)=O 55852,c1(OC)[nH]c(=N)ccc1C(N1CCN(C(C)CNC(C2(CO)CCC2)=O)CC1)=O 55853,N1(C(c2cnn(C)c2N)=O)CCC(CNC(c2cnc(C(F)F)s2)=O)C1(C)C 55854,CC1CN(C(=O)CC(F)F)CC(CCNC(=O)C(c2ccccc2F)(F)F)O1 55855,CCC(C)C(O)C(=O)N1CCCCC1CNC(C1(O)CC1)=O 55856,c1(CC)cc(C(=O)NC(C)CC(C)NC(c2cn(C)nc2C(C)C)=O)n(C)n1 55857,C#CC1(C(=O)NC(C)COCC)CCN(C(=O)C2=CCCSC2)CC1 55858,c1(C(C)=O)ccc(C)nc1NCC(CO)NC(C1CCOC(C)(C)C1)=O 55859,C1(C(=O)NCCCNC(=O)C(Cc2cccc(Cl)c2)=NO)CCC2CCC(=O)N12 55860,C1(F)(CNC(=O)CCF)CC2CCC(C1)N2C(=O)C=Cc1nccs1 55861,C(=O)(C(F)C(F)(F)F)N(C(CNC(c1cccc(CC)n1)=O)C)CC 55862,C(=O)(C1=NNC(=O)CC1)N(CC(CC)NC(c1ccc(Br)c(N)c1)=O)CC 55863,C=CCC(C(=O)NCCC1(CNC(=O)CN=S(C)(C)=O)CC1)C(C)(C)C 55864,CC1=C(C(=O)N2CC(NC(C3(C)CCCS3(=O)=O)=O)C(F)C2)SCCO1 55865,N1(C(C(CC)CO)=O)CCC(NC(C2(O)CCSC2)=O)C(C)C1 55866,[N-]=[N+]=NCC(C(=O)NC1CCN(CC2CCCCC2)CC1)NC(=O)OC(C)(C)C 55867,c1(NC(C2C3CN(C(c4occ(C(C)C)n4)=O)C2C3)=O)cnc(N(C)C)c(Cl)c1 55868,N1(C(C(CCC)C)=O)CCC2(CC1)CN(C(C1C=C1C)=O)C2C(C)C 55869,c1(OC)ccccc1CC(=O)N1CCC1CNC(c1oncc1C)=O 55870,c1(CC)cc(C(N2CCC(=CCNC(=O)C=CCN(C)C)CC2)=O)c(C)nn1 55871,CCC(CC)C(=O)NCC1CC(NC(c2cncc(C(=O)OC(C)(C)C)c2)=O)C1 55872,C1(CC(=O)NCCc2ncn(C)c2)COCCN1C(=O)Cc1cnn(C)c1 55873,C1(CC=C)(NC(c2cccc(C3CC3(F)F)c2)=O)CCN(C(C2CCSC2)=O)C1 55874,N1(C(c2cn(CC)nn2)=O)CCC2CN(C(=O)Cn3c(C)cc(O)cc3=O)CC12 55875,c1(C(=O)NC2CN(C(C3(C(C)(C)C)CCC3)=O)CC2F)ccc(=O)n(CCF)n1 55876,CC1(C)CC(c2ccccc2)(c2nnnn2C2CC2)N=C1C(=O)CC(C)(CO)OC 55877,C(CCCCC(=O)N1CC2CC(C1)C2NC(c1ncc(N)cc1Cl)=O)OC 55878,N1(C(C2N(C(C)=O)CC(O)C2)=O)CC2CCC2(NC(C2CC3CC3C2)=O)C1 55879,CC1(C)CCN(C(C2CCN(C(=O)CC3CCC(=O)N3)CC2)=O)CC1 55880,c1(CC(=O)N(C)CCNC(C2(Cc3cc[nH]c3)CC2)=O)ccc([N+](=O)[O-])cc1Cl 55881,C(C(=O)N1OC2CCC1CC2)N1CCN(C(=O)Cc2ccon2)CC1 55882,C(C)(CCCNC(C1(N(C)C(=O)OC(C)(C)C)CC1)=O)NC(CCSC)=O 55883,C(=O)(CC(CC)C(C)(C)C)NC(COCC)C(=O)NC1(CF)CC1 55884,CC1(C)C2CCC1(CC(N1CCN(C(=O)C(O)CC3CC3)CC1C(F)F)=O)CC2 55885,N1(C(C(CC)SC)=O)CCCCC(N(C(c2ccoc2C(F)(F)F)=O)CC)C1 55886,c1(NC(C2CC23CCN(C(=O)C=Cc2ccoc2)C3)=O)cc(I)ccc1CO 55887,N1(C(c2ccc(SCC)cc2)=O)CCC(C)C(NC(C23CCC(CC2)C3)=O)C1 55888,c1(C(=O)NC2C(C)CN(C(=O)C(c3ccnn3C)O)C2)nnn2c1CSCC2 55889,N1(C(c2ccnc(C)c2C)=O)CCOC2(CCN(C(c3[nH]cnc3C#N)=O)C2)C1 55890,N1(c2n(Cc3c(N=[N+]=[N-])cccc3)nnn2)CCCCCc2ccccc2C1 55891,C=CCC(CNC(=O)CCn1cncn1)C(=O)Nc1ccc(O)nc1 55892,c1(CNC2(CC(=O)Nc3ccnc(Cl)c3I)CCC2)c(Cl)[nH]c2ccccc12 55893,C1(C(N2CCC(CC(C)C)CC2)=O)CC2(CC2)CN1C(C1CC(OC2CC2)C1)=O 55894,c1(C(=O)NCC2CC(OC)CN2C(c2cnccc2Cl)=O)ccc(=O)n(C)n1 55895,CC(C)CCCC(=O)N1CC(O)CCC1C(=O)NCc1cccnn1 55896,Cc1cc(C(=O)NCCN(C(=O)COc2ccccc2Cl)C(C)C)c(C)n1C 55897,c1(C(=O)NC(C(C)C)(C)CNC(C2(O)CCSCC2)=O)ccn2cnnc2c1 55898,c1(CNC(c2c3c([nH]n2)C(C)CC3)=O)cc2c(cc1O)OCO2 55899,c1(N(CC(C)OC)C)nc(N2CCCN(CCO)CC2)nc2sccc12 55900,C(=O)(CCCCC(N)=O)N1CCCC(NC(COc2c(C)cccc2Cl)=O)CC1 55901,C(C(CC(F)(F)F)NC(C1(CC)CC1(F)F)=O)NC(c1cnc(OCC)nc1)=O 55902,C(C)(CN(C)C)(C(=O)N1CC(N2CCCC2)C1)NC(c1cnn(C(C)C)n1)=O 55903,C1(CNC(C2CCCC2c2nc[nH]n2)=O)CCCCN1C(c1ccsc1Cl)=O 55904,Cc1coc(C)c1C=CC(=O)NC(C1CCCN(C(C2CC(F)(CO)C2)=O)C1)C 55905,C1(NC(=O)C=Cc2ccc[nH]2)COC2(CNC(=O)C(=Cc3cccs3)F)CC1C2 55906,c1(OCC)nc(C(=O)NC(C)C(C)NC(c2ccn(C3CCOCC3)n2)=O)ns1 55907,c1(CCC(=O)NC(C2CN(C(CCNC(=O)NC)=O)C2)C)cccc(F)c1 55908,c1(C(N2CCC(C(C)(C)NC(c3coc(O)n3)=O)C2)=O)cc(Cl)cc([N+](=O)[O-])c1 55909,N1(C(C(CC)(C)OC)=O)CCC(C2CCN(C(c3c(C)noc3C)=O)C2)CC1 55910,C1(F)(C(=O)NCCCCNC(C2(c3ccno3)CCC2)=O)C2CCCC12 55911,C12(CNC(C(C)C3CCOC3)=O)CC(CO1)N(C(c1scnc1Cl)=O)C2 55912,C(=O)(CCC(C)CN(C)C)NC(C(N1C(C)(C(=O)NC)CCC1)=O)C 55913,CC1(C)CCCN(C(c2cncs2)=O)C1C(=O)NC(CCO)C1CC1 55914,C#CCCN=C(NCc1cnccc1O)NC(C)CCc1ccco1 55915,c1(C(N2C(CNC(C3(C)CCOC3)=O)CC2)=O)ccc(Cl)cc1C(=O)O 55916,C1(C2CC2)(C(N2CCC(NC(c3sccc3F)=O)CC2)=O)CC=CC1 55917,Cn1nnc2cc(C(N3CCCC(NC(=O)C4=CC(C)(C)C4)C3)=O)ccc12 55918,C(=O)(C(CNC(=O)CCC1CC1(F)F)CC(C)C)NCCc1ccc(C)s1 55919,C(=O)(C(CO)C(C)(C)C)NCC(CCC)C(=O)NCc1cccnn1 55920,N1(C(C(=O)Nc2cccc(C)c2)=O)CCN(C(=O)Cc2cnc(C)s2)C(C)C1C 55921,Cc1cc(F)ccc1CNC(=O)C(c1ccncc1)N1CCCC1C1CCCC1 55922,C12(C(=O)NCC(C)N(C(=O)Cc3cnns3)CC)CCCC1CCC2 55923,c1(CNC(=O)Cc2cnoc2)ccnc(C(=O)NC2CCS(=O)CC2)c1 55924,C(CN=C(NCCCCN1CCCCCC1)NCC1CCCCO1)=CC=CC 55925,N1(C(C(C)n2cncn2)=O)CCOCC1CN(C)C(c1nccnc1C(N)=O)=O 55926,c1(C(=O)NC(CN(C(C2(CC(=O)OC)CC2)=O)C)C)ccc(-c2ccncc2)o1 55927,O=C1CN(CC2CC2(Cl)Cl)C(=O)N1CCC1(C(F)(F)F)CC1 55928,CC(C)C(C(=O)NCCCCCNC(c1ccccn1)=O)SCc1ccccc1 55929,C1(CCNC(C(C=C)(C)O)=O)CN(C(=O)C(C)OC2CCOC2)CCCO1 55930,N1(C(CC(=C=C)C)=O)CC2(CCN2C(c2ccc(OC(C)=O)cc2)=O)C1 55931,C1(CNC(C(Cn2ccc(C)n2)C)=O)CCN(C(=O)C(C)(C)NS(C)(=O)=O)CC1 55932,CCC(C)CC(C)C(=O)NC(CNC(c1ccccc1CO)=O)(CC)CC 55933,c1(NC2C=CC(C(=O)NCc3ccc(C)c(Cl)c3)C2)ccnc2ccnn12 55934,N1(C(C=Cc2cn(C)nn2)=O)CCCN(C(c2nn[nH]c2Cl)=O)CC1 55935,N1(C(c2c(C)cn(C)c2)=O)CCCC(O)(CCNC(=O)C=C2CCC(C)C2)C1 55936,C12(CNC(CC(=O)NCC#C)=O)CCCC1CN(C(=O)C(F)(F)CCC=C)C2 55937,C(N=c1ccnc(NC2CCC2C2CC(C)(C)CCO2)[nH]1)c1ccc(C)c(Br)c1 55938,C1(C#N)(C(=O)NCCN(C(C2CCCS2)=O)CC)CC1 55939,c1(C(=O)NCc2n(C)nnc2-c2ccccc2)ccc2c(c1)CC(O)C2 55940,C(N=c1[nH]cnc2[nH]cc(CO)c12)C1CCCN(C(c2ccc(F)s2)=O)C1 55941,C=C=CC(C)C(=O)N1CCC(OCCNC(C2CCC(=O)N2CC)=O)C1 55942,Cc1nn(CC(=O)NC2CC(NC(=O)C(C)CN(C)C)C(O)C2)c(C)c1[N+](=O)[O-] 55943,c1(NC2C(C)COCC2)[nH]c(=NCc2sncc2Br)nc2c1ncn2C 55944,c1(C(N2CCCC(CCNC(CC(C)F)=O)C2)=O)ccn2ncccc12 55945,CC(C)(CNC(=O)C=CCO)CC1CN(C(c2cnc(C(F)F)s2)=O)C1 55946,CCCCCC(=O)NC1COCCC1NC(c1cnc(C2CC2)[nH]1)=O 55947,C1(CC(N2CCC(O)(CN(C(C3CC(OC)C3)=O)C)C2)=O)CC2(CCC2)CO1 55948,c1(C(N(C(=O)Cn2cc(C(=O)OC)nn2)CCOC)C)cccnc1O 55949,C1(CC=C)(NC(c2cnn(C)c2OC)=O)CCN(C(=O)CC2CC2C)C1 55950,C(=O)(C1=NOC(C)C1C)NC(C1N(C(c2ccc(OC)cc2OC)=O)CCC1)C 55951,C(CC(C)(C)C)(C(=O)NCCC1CC(C(=O)N(C)Cc2cn(C)cn2)C1)OC 55952,c1(C(N(C)Cc2ccc(C)cc2Br)=O)n[nH]c2cccc(F)c12 55953,C1(NC(c2cn(C)nc2Cc2ccccc2)=O)CN(C(=O)C=CCF)CCC1F 55954,Cc1ccc(C=CC(N2CCC(NC(=O)CC3(C)CCCO3)CC2)=O)s1 55955,C(CN=c1[nH]c(=NC2CCC(C3CC3)CC2)[nH]c2c1SCC2)C1(OC)CCC1 55956,C1(C(N(CCCNC(c2ccnc(OC)c2F)=O)C)=O)COc2ccccc2O1 55957,CN1C(=O)CCC1CC(=O)NC1CC(CC(=O)NCC(F)F)C1 55958,CC(C(=O)N1CCCC(NC(c2cnc(N)c(CO)c2)=O)C1)C(C)(F)F 55959,C(C(=O)N(CCCNC(=O)CO)C(C)C)(C1CC1)SC 55960,C1(C)(C(=O)NC2CN(C(C(c3ccc(F)cc3)(C)F)=O)C2)CC(C2CC2)=NO1 55961,N1(C(C(CC=C)C(=C)C)=O)CCC2(CCC2C(=O)NCc2cc(Cl)ccn2)CC1 55962,c1(C(=O)NCC(CCCC)NC(=O)C(O)C(C)(C)CC)cccc2ccncc12 55963,Cc1c(C(=O)NC(C)C(C)CN(C)C)ccn1CCO 55964,c1(C(N2C(CNC(CC(C)N(C)C)=O)CC3(CC3)C2)=O)cccc2nccn12 55965,C1(NC(c2c(C)cc[nH]2)=O)CN(C(=O)Cc2ccccc2CS(N)(=O)=O)CC1O 55966,N1(CC)CCOC(C)(CNC(=O)CC(c2cccs2)NC(C2(Br)CC2)=O)C1 55967,N1(CC(=O)NC(CC)CNC(=O)C(F)(F)c2cnnn2C)CCN(C)C(=O)C1 55968,N1(C(COC)=O)CC2(CCN(C(=O)CC3CC(O)C3(C)C)CC2)CC1C 55969,N1(C(c2cccc(C(=O)OC)c2)=O)CCC(C)(CNc2ccc(I)cc2Br)CC1 55970,c1(CCC(C)=O)nc(-c2ccnc(N3CCCCC3)c2)nn1CC(C)O 55971,C(C)(C(CC(=O)NCCC(C(C)C)OC)NC(C1CN2CCC1CC2)=O)OC 55972,Cc1cnc(CC(=O)N(C2CCN(C(C3CCSC3)=O)C2)CCO)s1 55973,N1(C(C2CC=C(C)CC2)=O)CCCC(CCNC(=O)C=CC(C)C)CC1 55974,C1(C(=O)NCCN(CCOC)C)CC2(CC(NC(=O)C(c3c(C)n[nH]c3C)C)C2)C1 55975,C1(C(C)NC(=O)C(F)Cc2ccccc2)CN(C(c2cnoc2)=O)CCO1 55976,C(CC(C(=O)NCCC(C1CC1)C1CC1)NC(=O)CSC(C)(C)C)OC 55977,Cc1c(C(N2CCOC(CC(=O)N(C3CN4CCC3CC4)C)C2)=O)c[nH]c1C#N 55978,Cc1c(C(N2CCC(CN(C(=O)C(C)NC(C)(C)C)C)C2)=O)sc(Cl)c1Cl 55979,C1(C(=O)NC(CC)CSC)CN(C(c2ccc(CO)cc2)=O)CC(C)(C)C1 55980,C1(O)(CCNC(C(C)(C)C2CC2)=O)CCN(C(=O)CC(=O)NCC2CC2)C1 55981,c1(C(=O)NCCN(C(C2CC3OC(=O)OC3C2)=O)CC)nn(C)c2c1CCC2 55982,C1(NC(c2occ(C)c2)=O)CCCCC12CCN(C(c1cnc(F)c(C)c1)=O)C2 55983,C(=O)(C1=NOC(C)C1C)NCC(C)NC(C1(C(C)C)CCC1)=O 55984,N1(C(c2c(C)nc(O)cc2)=O)CC(CNC(=O)C(C)n2cnnn2)CC(C)(C)C1 55985,C1(NC(C(C)NC(N)=O)=O)CCC(N(C(=O)Cn2cnc(Br)n2)C)CC1 55986,N#Cc1ccc(CN2CCCC(NC(c3ccnnc3O)=O)C2)c(Br)c1 55987,c1(N(CCOC)C(c2ccc(Cl)c(Cl)c2)=O)nc2ccccc2s1 55988,N1(C(c2ccc(C)c(C)c2)=O)CCC(NC(c2cnc[nH]2)=O)C(CO)CC1 55989,C1(NC(c2n(CC)nc(C)c2)=O)C2CCC1N(C(=O)CN1CC3CC3C1)C2 55990,CN1CC(C(=O)NC2(C(=O)NCC3(CO)CCCCC3)CCSC2)CCC1=O 55991,N1(C(C(C)(C)OC)=O)CCCC(CCNC(c2ccc(C)nn2)=O)CC1 55992,c1(CC(=O)NCCC(=C)CNC(C2CCC(C)=C(C)C2)=O)cccc(O)c1F 55993,C1(C=O)C2CN(Cn3cc(C4CC(CO)C4)nn3)CC12.C1(OCC)CCCOC1 55994,N1(C(c2ccnc(OC)n2)=O)CCC(C)N(C(c2ccncc2C)=O)CC1 55995,c1(C(N(C(CNC(c2cc(C(=O)OC)no2)=O)C)C)=O)noc2c1COCC2 55996,C1(CC(=O)NC(CCC)CO)CN(C(=O)Cc2ccsc2)CCC1C 55997,C(=O)(CC(CCC)NC(C1(C2(C)CC2)CC1)=O)N1CCC(C=C)C1 55998,C1(CC#C)(C(=O)NCCC(C)N2CCCC2)CCN(C(C2CC2(F)Br)=O)C1 55999,C1(C(F)(F)F)(C(N2CC(CC(C)NC(=O)CCc3cncs3)C2)=O)CCCC1 56000,C1(CO)CN(N2CC3CCCC(C3)C2)CC12CCOCC2 56001,N1(C(C2(C)CC(C)(C)C2)=O)CCN(C(C2C=CCCC2)=O)C(CC(F)(F)F)C1 56002,c1(C(=O)NCc2cn(CCNC(CC=CC=C)=O)nn2)ccccc1C 56003,N1(C(c2ccc(C#C)c(F)c2)=O)CC2C3CCC(C2C1)N(C(=O)C(CC)CC)C3 56004,n1(C(C)C)ccc(=NC(=O)CCC(C)NC(=O)C(c2ccn(C)n2)C)[nH]1 56005,C1(NC(CC2CC(C)NC2)=O)CCC2(CCC2)C1 56006,n1(C(C)C)cnc(C(=O)N(CCNC(C2CC2(C)C(C)C)=O)C2CC2)c1 56007,N(C=CC(=O)C(F)(F)F)C(C1N(C(c2cccc(I)c2)=O)CC(O)C1)=O 56008,C12(CS(=O)(=O)CC3(NCc4c(C)ccc(N)c4)CC3)CCC(C(=O)O)(CC1)CO2 56009,c1(C(N2CC=CC(NC(C3C(C)(C)C3)=O)C2)=O)cnc2ccccc2c1 56010,C1(NC(C2CCC3(CC2)CC3)=O)CS(=O)(=O)C12CCN(C(=O)CCC(F)F)CC2 56011,CC1(C)C(C(F)F)CCN1C(c1cc(C(F)F)ncn1)=O 56012,N1(C(CCCOCC=C)=O)CCN(CC(=O)NCCCC(O)CO)CC1 56013,N1(CC(=O)NCC(C(C)C)NC(C2CCCC2C(F)(F)F)=O)CCS(=O)(=O)CC1 56014,CCCCC(C)(F)C(=O)N1CCC(O)(CNC(C2(C)CCCC2)=O)C1 56015,c1(-c2cc(N(CC)CC)ncc2)c[nH]c2cc(C(=O)NCCSC)ccc12 56016,C(=O)(C(C)S(N)(=O)=O)NCC1(C(N)=O)CN(C(c2c(C)cc(SC)o2)=O)C1 56017,c1(C(=O)NC(CN(C(Cc2cc(CC)on2)=O)C)C)ccnc(OCCN(C)C)c1 56018,C1(CN(C(C2C(C=C(C)C)C2(C)C)=O)CC)CCCCN1C(c1n[nH]cc1Cl)=O 56019,CCC(CC(=O)NCC(CO)NC(c1cnc(C2CC2)s1)=O)C1CC1 56020,N1(C2CCN(C(C(C3CCCCC3)=O)=O)C2)CCN(C(=O)CCC2CCC2)CC1 56021,c1(NC(C(=O)NCC(c2cccs2)=O)=O)ccc(I)c(Br)c1Cl 56022,C=C1CC2CCC(C1)N2C(=O)C(F)C(C)CNC(C1(C(N)=O)CCC1)=O 56023,c1(C(=O)NC2CC(OC)CN2C(c2ccc[nH]2)=O)ccc2[nH]c(C(N)=O)cc2c1 56024,C1(CNC(C2(OC)CCC2)=O)CCN(C(c2cccc(=O)n2C)=O)C12CC2 56025,C1(O)(CC(N2C(C)(CC(=O)NCCc3ccc(O)nc3)CC2)=O)CCCCCC1 56026,c1(NC(N2CCCC(n3ccnc3)C2)=O)ccc(-c2ncc(C(F)(F)F)s2)cc1 56027,CCC(C)C(C(=O)NC1CC(C)(NC(=O)CCNS(=O)(=O)c2cccs2)C1)OC 56028,C1(C(N2CCC(CC=C)(NC(c3sc(F)cc3C)=O)C2)=O)C2CCCCCC12 56029,C1(NC(Cc2n(C)ncc2)=O)CC2CCC(C1)N2C(c1c[nH]c2nccc-2c1)=O 56030,c1(C(N2CCCC2Cc2ccccc2)=O)ccc(C(F)C(F)(F)F)nc1 56031,c1(C(=O)NC2(C)CC(NC(C=CC=CCC)=O)C2)c(C)nn(C)c1Cl 56032,C=C(C)CN=C(NCC1COCC(C)(C)O1)N1CCC(F)(F)C(C)C1 56033,C1(CC(=O)NC(CNC(C=CC)=O)C2CC2)CC(=O)c2ccccc2C1 56034,c1(C(=O)NCC23N(C(C=C4CCC(C)C4)=O)CC(C2)C3)cc2c(s1)CCC2 56035,c1(C(N2C3C(NC(c4c(COC)ccs4)=O)CC(C3)C2)=O)nccc2n[nH]cc12 56036,C(c1ccc(O)cc1)=CC(=O)NC1(CO)CCN(C(C=CCN(C)CC)=O)C1 56037,C1(NC(C(COC(C)C)NC(c2ccc(CC)o2)=O)=O)COCC1C1CC1 56038,c1(C(=O)NC2CCC(NC(C(CC=CCC)C)=O)CC2)c(C)nn(CC)c1Cl 56039,C1(CN(C(=O)Cc2cccs2)C)CN(C(=O)CCNC(C2CCC2)=O)CCO1 56040,C(=O)(CC(O)C(C)C)NCC1(OC)CN(C(c2ccnc(-n3cccn3)c2)=O)C1 56041,Cc1nsc(C(N2CCC3C(NC(c4ccnc(S)c4)=O)C23)=O)c1N 56042,c1(COC)ccnc(C(=O)NC(C2CCOC2)CNC(=O)CP(C)(C)=O)c1 56043,C(=O)(C(O)(C(F)(F)F)C1CC1)NCC1(C)CC=CC1 56044,C1(C(=O)NCC(C(C)C)(C)NC(=O)C(C)CO)CCC(F)(F)CC1 56045,C1(CNC(c2c(C)nc(C)s2)=O)CC(C(C)(C)C)CN(C(=O)Cc2cnoc2)C1 56046,C1(CC=C)(C(=O)NC2CCN(C(=O)Cn3cc(C#N)cn3)C2CC)CCCCC1 56047,CCC(C(=O)NCC1CCCC1NC(=O)C(C)(C)F)NC(N)=O 56048,C1(C(=O)NCC2(NC(C(C(C)C)OC)=O)CCCC2)CCC(F)(F)CO1 56049,C(=O)(C1=Cc2ccccc2C1O)NCC1CCCN(C(C=NOC)=O)C1 56050,CCS(=O)(=O)CCCN=C(NCC1CCOCC12CCC2)NC1CCC1 56051,C(C(=O)NCC(C)N(C(=O)CCc1cnn(C)c1C)CC)(C(C)C)OCC 56052,CCCCCC(O)C(=O)N(c1ccc(F)cc1C)C(C1C(N)C2CCCCC12)=O 56053,N1(C(CCC(C)OCC)=O)CCC(C)(C)C(NC(c2cc(C(F)(F)F)no2)=O)C1 56054,Cc1nc2cccc(C(N3CCN(C(C4COC(=O)O4)=O)C(C4CC4)C3)=O)c2[nH]1 56055,N1(CC)CCC(C(=O)NC(C)(CSC)C(=O)N(CCCC(C)C)C)CC1 56056,C1(C(C)OC)CCCN(C(=O)CCN(c2cc(C)co2)C(c2cccs2)=O)C1 56057,c1(CNC(C2CCC(C)(CC)O2)=O)nc2c(s1)CN(C(=O)COC(C)(C)C)CC2 56058,N1(C(C(CC)c2cccnc2)=O)CC2CN(C(=O)Cn3c(C)ccc3C)CCC12 56059,C1(O)(C(=O)NCC(C)NC(c2ccc(CO)o2)=O)CCCC(C)(C)CC1 56060,N1(C(C2(COC)COC2)=O)CC(C)CN(C(=O)Cc2c[nH]nc2C)C(C)C1 56061,C1(C2CCCO2)(NCc2nnn(C(C)(C)C)n2)CSC(C(C)(C)C)C1 56062,C(=O)(N=S(C)(=O)CCO)NC(CC)Cc1ccc(Cl)cc1 56063,c1(-c2c(C(=O)NCC(CC)NC(C3COCCN3C)=O)c[nH]n2)cccc(Cl)c1 56064,c1(CC)occc1C(N1CCCC1C1CCN(C(c2cc(C3CC3)no2)=O)C1)=O 56065,C(=O)(CC1=CCOCC1)N1CCC(CNC(c2c(Cl)c(C)n(C)n2)=O)C(C)C1 56066,C(=O)(CCCC(CC)NC(=O)CCCCCC)NC(C1CCOC1)C#C 56067,N1(C(C(CC)F)=O)CC2C(CNC(=O)CCc3nnc(C(F)F)o3)C2C1 56068,N1(C(CC=CC=C)=O)CCC2CCN(C(c3cc(C(N)=O)co3)=O)C2C1 56069,N1(C(C(Cc2ccc(C)cc2)C)=O)CCN(C(c2ccc(=O)n(C)c2)=O)CC1C 56070,Cc1cc(N)c(C)nc1C(=O)NCCCNC(=O)C=CC1CC1 56071,c1(-c2ccc(OCC)cc2F)nc2ccc(C(N3CCC(C(N)=O)C3)=O)cc2s1 56072,NS(=O)(=O)c1cncc(C(=O)NC23CC2CN(C(C2CCCCC2)=O)C3)c1 56073,N1(CC)CC(C(=O)NC2CCC(CNC(=O)C(F)(F)CN(C)C)CC2)CC1=O 56074,N1(C(CCC#C)=O)CCC(C)C1CNC(=O)CCSc1nnnn1C 56075,CON(C)C(=O)c1conc1CNC(=O)Cn1cnnc1 56076,C(CS(=O)(=O)CCCN1CCCC(NC(=O)C(c2ccccc2)O)CC1)OC 56077,C1(NC(c2cncnc2)=O)CN(C(=O)CCN2C(=O)CCC2=O)C2(CCOC2)C1 56078,c1(SC)cccc(CC(=O)NCC2(O)CCN(C(C3(c4nccs4)CC3)=O)C2)c1 56079,C1(C(N(C)CC2(O)CN(C(=O)CN3CCSCC3)C2)=O)SC2C=CC1CC2 56080,C1(C(=O)NCCC(CNC(CCCN(C)C)=O)O)OCCOC12CCC2 56081,Cc1coc(C2CC2)c1C(=O)NCCCCNC(C12CCCCC1C2)=O 56082,Cc1cc(C(c2nnnn2CC2CCCO2)Nc2cnoc2)c(Br)cc1F 56083,c1(C(N2CC(SC)C(NC(=O)CCC3CC(F)(F)C3)C2)=O)n[nH]c2c1CSCC2 56084,N1(C(=O)OC(C)(C)C)CCC(NS(=O)(=O)NCC2CC2c2ccncc2)CC1 56085,C1(CNC(C(CC)OC)=O)CC2(CCN(C(=O)C(O)CCSC)C2)CO1 56086,C#CC1CCN1C(=O)C(Cn1ccnn1)NC(=O)C(C)=CC(C)(C)C 56087,CCC(CCC(=O)Nc1ccccc1CCO)NC(C1CCCCC1O)=O 56088,C1(NC(C2CC2[N+](=O)[O-])=O)CC2C1CCN2NC(c1ccnc(S)c1)=O 56089,N1(C(=O)COCC(F)F)CCC(O)(CCNC(C2(c3ccc(F)cn3)CC2)=O)C1 56090,N1(C(=O)C(O)Cc2cnc[nH]2)CCN(C(c2cnccc2Cl)=O)C2COCC12 56091,N1(C(CC(=O)NC)=O)CCC2(CC1)CC(NC(=O)CNC(c1cccc(O)c1)=O)C2 56092,C1(C)(NC(CCOCCC)=O)CCCN(C(c2[nH][nH]c(=N)c2Br)=O)C1 56093,C(CCN(C)C)(C(=O)NC1CCCCC1)NCc1nc(NC(C)=O)sc1 56094,CC(C)C(C)(O)CNC(c1cc(NC(C2(n3nccn3)CC2)=O)nn1C)=O 56095,CC1CN(C(c2ccnc(Cl)c2)=O)CCC1N(C)C(c1cc(=O)cc[nH]1)=O 56096,C1(C(=O)OC)CCC(C(N2CCC(CCNC(=O)CC=C(C)C)C2)=O)CC1 56097,N1(C(=O)C(Cl)=CCl)CC2CC1CN2C(C1(C(=O)NC2CC2)CC1)=O 56098,N1(C(c2c(CC)nco2)=O)CC(C)OC2(CCN(C(=O)CSCC(C)C)C2)C1 56099,c1(CC=C)ccccc1C(N1CCC(N(C(C2COCCN2CC)=O)CC)C1)=O 56100,C1(F)(CNC(Cc2ccn(C)n2)=O)CCN(C(C2CC(N3CC(O)C3)C2)=O)CC1 56101,C1(NC(=O)CSCc2cccnc2)COC2(CCN(C(c3ccc(F)o3)=O)C2)C1 56102,C(N1CCC(F)(F)CC1C)c1n(CCC(CC)(F)F)nc(-c2ccc(Cl)cn2)n1 56103,c1(C(c2cnc(N3C(C)(C(=O)O)CCCC3)s2)=O)ccc2nc[nH]c2c1 56104,CCC(O)C(C)C(=O)NC12CC(C(N3CC(c4ncc(C)o4)C3)=O)(C1)C2 56105,C1(O)(CC)CCN(C(=O)C(C)(C)CN(C(=O)CCC(C)SC)C)C1 56106,N1(C(C(C)(C)S(C)(=O)=O)=O)CCC2(COCC(CNC(=O)Cn3cnnn3)O2)C1 56107,Cc1ncc2n1CC(C(=O)NC1CN(C(C3CCOC(C)(C)C3)=O)CC1C)CC2 56108,N1(C(CC(COC)COC)=O)CCCC2(CCC2NC(=O)CC2CCC2C)C1 56109,C1(CCC(=O)NCC(CC)(C)NC(=O)COC(C)C)CCC(O)CC1 56110,N(C(=NCC=C1CCOCC1)N1CCC(c2nncs2)C1)CCOC(C)(C)C 56111,c1(NC(=O)OC)cccc(C(=O)NC(C)C(C)NC(C2(C)CCCC2C)=O)c1 56112,S(=O)(=O)(c1ccc(F)cc1Cl)NC(c1ccc(S(C)(=O)=O)cc1)C 56113,N1(C(C2C(OC)C2)=O)CCC(C)C(CNC(=O)C=CC=C(Cl)Cl)C1 56114,C1(CC(=O)N(CCOCCCN(C(CCOCCOC)=O)C)C)CCCC12CC2 56115,c1(C(=O)OC)c(Cl)nc[nH]c1=NCCCN(C(=O)C1=CCCCO1)C 56116,C1(CC)C(C(=O)NC(CCSC)C(=O)NC(C2(CO)CC2)C)CCN1C 56117,Cc1ccn(C(C)CC(=O)NCC2(C)CC(NC(c3cc(F)cs3)=O)C2)n1 56118,N1(C(CC(C(C)OC)NC(c2cc3n(n2)CCC3)=O)=O)CC(C)NC(=O)C12CC2 56119,C#CCCC(O)C(=O)NCC12CC1CN(C(=O)Cc1cccc(Cl)c1F)C2 56120,C1(CNC(C2C(C(C)NC(Cc3c(C)n[nH]c3)=O)C2)=O)CC2(CCC2O)C1 56121,c1(C(N2C(C(N3CCn4cccc4C3)=O)CC(C)C2)=O)ccc([N+](=O)[O-])cc1I 56122,CCCC(C(=O)NCC(C)(C)CNC(c1cc(Br)cc(N)c1C)=O)C(C)C 56123,CC1=C(C(=O)N2CCC(C3(NC(c4sccc4F)=O)CC3)C2)CCCC1 56124,c1(C(N(C(CNC(C=C(C)C(C)C)=O)C)C)=O)cc(F)cc(Cl)c1O 56125,C(c1cc(C)cc(C)c1)=CC(N1CC(NC(c2cccc(OC)c2F)=O)C1)=O 56126,N1(CC(=O)NCCc2ncoc2C2CCC2)CCCCC1 56127,CCCCC(COCCNC(=O)NC12CC3CC1C2C3)CC 56128,c1(CC(N2CC(O)C23CCOCC3)=O)ccc2ccccc2c1Br 56129,C1(NC(C2CC3CCC2O3)=O)C=CCN(C(=O)CCc2ccco2)C1 56130,CC1(C)CC(NC(c2ccc(-c3ccon3)cc2)=O)CN(C(=O)COC2CC2)C1 56131,c1(CCC(=O)NC(CNC(CCOCC(C)C)=O)(C)C)cc(Cl)no1 56132,N1(C(C2(CC#C)CCCO2)=O)CCCC(C)(NC(c2cc(O)nc(O)n2)=O)C1 56133,c1(NC(C)=O)ccc(-c2csc(NC(c3cc(Cl)c(Cl)s3)=O)n2)cn1 56134,CC(CC(C)(C)C)C(=O)NCCOCCCNC(=O)CSc1nncn1C 56135,c1(C(=O)NC(CCC)CNC(C2CC=CCC2)=O)cnc2ncccn12 56136,c1(C(=O)Nc2cccc(C(N=c3nc(C)[nH]s3)=O)c2)ccc2c(c1)CCCCN2 56137,N1(C(C(C)SC2CC2)=O)CC2CC1CCC2NC(c1ccc(OC(C)C)nc1)=O 56138,Cc1c(Cl)c(C(N2CC(CNC(=O)Cc3cccnc3Cl)CC2C)=O)nn1C 56139,C(=O)(CCCCC(F)F)NC(C)C(CO)NC(=O)Cc1cnccn1 56140,N1(CCC(=O)NCCNC(C(CC)F)=O)CCCCCC1 56141,c1(OC)ccc2c(c1)C(NC(=O)C(N1c3ccccc3CCC1C)=O)CC2 56142,c1(CN(CC(C)NC(C2CCN(C)C2=O)=O)C)cccc2nsnc12 56143,C(=O)(CCc1ccsc1)NCCN(C(=O)COC)CCC.C1(=O)CCN1 56144,Cc1nc(C)c(C(N2CC(NC(c3ccnn3C(F)F)=O)C(C)(C)C2)=O)nc1C 56145,CC(C)C(CNC(=O)CCCSC(C)(C)C)NC(=O)Cc1cnn(C(F)F)c1 56146,Cn1cc(S(N)(=O)=O)cc1C(=O)C(=O)NCCC1CCCCN1C(=O)CC(F)F 56147,c1(OCC(=O)NC2CC(C)N(C(C3CC4CC3C3CC43)=O)C2)ccccc1C#N 56148,CCCCC(O)C(C)C(=O)NC(c1cnn(C)c1)C(=O)NC(C1CCOC1)CO 56149,c1(C(N(C2CN(C(Cc3cnc(C)o3)=O)CC23CC3)C)=O)ccn2cccc2c1 56150,C12(CNC(c3cc4n(n3)CCC4)=O)CCC(CC1)N(C(C1CCCC(CF)C1)=O)C2 56151,Cc1cccc(CC(=O)NC2CC2NC(=O)C(C)C2CCCC2)c1 56152,N1(C(Cc2n(C)nnc2)=O)CCC2(CCOC2)C(CNC(C2(CCO)CC2)=O)C1 56153,C(N=C(NCC(F)F)NC1CCN(C2CCCC2)CC1)C1C(OC)CCC1 56154,C1(C(=O)NCc2ccc(N(C)CC)cc2)CC2CCCC2C1 56155,N1(C(C2C(CCOC)C2)=O)CC(NC(=O)Cn2cc(Cl)cn2)C(CC2CC2)C1 56156,C1(NC(CC(CC)CC)=O)CC2CC1CN(C(c1ccc3nncn3c1)=O)C2 56157,C1(NC(c2ccccc2Cl)=O)CN(C(C2CCC3(CCC3)OC2)=O)CC2(CC2)C1 56158,Cc1c(C(=O)NC2CCCC(NC(=O)C(F)=C3CCCC3)C2)sc2ccccc12 56159,c1(C(N2CCN(CCNC(CCCSC)=O)CC2)=O)ccnc2ccc(O)cc12 56160,N1(C(CC#C)=O)CC2CCCC2(NC(=O)Cc2cc(OC)cc(Cl)c2)C1 56161,O=C(C#CC1CC1)N1CCC(C2CCCN2C(c2cc(=O)cc[nH]2)=O)C1 56162,C1(C(=O)NC(Cc2cn(CCOC)nn2)C(=O)OC)CCC2(CC1)CC(O)C2 56163,C1(C(=O)NC2CCN(C(CC)=O)C2)CN(C(C23C=CC(CC2)C3)=O)CC1F 56164,C(=O)(CCCCC#N)NCCC1CC(NC(C2(C)COCCO2)=O)C1 56165,N1(C(c2c(CC)cncc2)=O)CC(C(=O)NC(c2n[nH]c(CO)n2)C)CC(C)C1 56166,C1(C#N)(NCCNC(CCCC(=O)N(C)C)=O)CC2C=CC1C2 56167,C(CN=c1[nH]c(=NCc2cc(C3CC3)n[nH]2)[nH]c2cccc(F)c12)SC(F)(F)F 56168,c1(C(=O)NC2C3CN(C(c4ccc(SC)s4)=O)CC32)ncc2c(F)cccn12 56169,C=CCCC(C(=O)NCc1ncc(CO)[nH]1)NC(=O)C=CCc1csnc1OC 56170,C1(NC(C2C(C)(C)C2)=O)CCCCCC1C(N1CC(OCF)C1)=O 56171,C1(CN(C(c2c(C)nsc2)=O)C)CCCC(NC(c2cc[nH]n2)=O)C1 56172,C1(NC(c2ccc(CSC)o2)=O)CC2CCC1N(C(=O)C(C)n1cnnn1)C2 56173,C(=O)(CC(C(F)(F)F)n1cccn1)N1CCC(Sc2cc(C(C)=O)nn2C)CC1 56174,C1(C(=O)NC2(C#C)CCOC2)CCC2(CC2)N1C(C1CN2CCN1CC2)=O 56175,c1(OC)ccc(CCC(N2CC=CC2CNC(C2CCCO2)=O)=O)cn1 56176,N1(C(c2cc(OC)ns2)=O)CC(C(N2CCNC(=O)C2C(C)C)=O)CC(C)(C)C1 56177,Cc1cccc(Br)c1C(C(=O)NC1(C)CC(C)OC1=O)NC(c1cc(Cl)ns1)=O 56178,C=CC(C)(O)C(=O)NCC(c1ccco1)NC(c1csc(-c2cocn2)n1)=O 56179,CN1CCOc2c(C(N3CC(NC(=O)C(O)C(F)(F)F)C3)=O)cccc21 56180,c1(C(=O)NCC(C2CCC2)NC(C2C(CC(C)C)C2)=O)nsnc1O 56181,C12CN(C1)C2=O.C1(CCOC)(C(=O)NCC2CC(C(=O)OC)C2)CCC1 56182,C(C)(C)(CCCCC(=O)NC1CCN(C(c2ccc(Cl)c(Cl)c2)=O)CC1)OC 56183,Cc1cnnc(O)c1C(=O)NCc1cc(C(N2CCC(C)C2CO)=O)no1 56184,CC(CN=c1nc(N2CC3C(C)C3C2)c2c([nH]1)CCCC2)N(c1ccccc1)C 56185,C1(NC(c2cn(CCOC)nn2)=O)CC(NC(C2C=CCS2)=O)C12CCC2 56186,c1(C(N2CC3C(CN(C(C(C=C)O)=O)C)C3C2)=O)cc(C)cc(C)c1 56187,CCCCC(C)(C)NC(=O)C(Cc1ccc(C)cc1)c1ccccc1 56188,CC1CC=C(C(=O)NCC2CCC2NC(=O)CSc2nnnn2C2CC2)CC1 56189,Cc1ccc2c(CC(N3CCN(C(C45CC(C)(C4)C5)=O)CC3)=O)c[nH]c2c1 56190,c1(CNC(C(C)c2cccs2)=O)ccoc1C(=O)NCc1ccnn1C 56191,C(C1=C(C(=O)O)C(c2ccccc2)NC(=O)N1)N(C(=O)C1=NNC(C(F)(F)F)C1)C 56192,N1(C(C(C(=O)OCC)(C)C)=O)Cc2occ(C(=O)NCCCSCC)c2C1 56193,N1(C(C2C(C)CCC2)=O)CCC2(CC(NC(c3cccs3)=O)C2)C1 56194,CC1CN(C(c2cn(CCNC(=O)CC3CCCC(=O)N3)nn2)=O)CC(=O)N1 56195,C(=O)(C(C)(C)CCCCC)NC1CN(C(C2(CC#C)CC2)=O)CC(C)C1 56196,C1(NC(c2cc(CSCC)on2)=O)CC2CC1N(C(=O)C(C)(C)CN(C)C)C2 56197,N1(C(C2(F)CCN(C(c3cc(C)ncc3C)=O)C2)=O)CCCC12CCCOC2 56198,N1(C(CSS(C)(=O)=O)=O)CCOCC1C1CC(F)C1 56199,c1(C(N2CCC(CC3CN(C(c4cnco4)=O)C3)CC2)=O)ccn2ccnc2c1 56200,c1(C(N2CCC(N(C(=O)C(C)CF)CC)C2)=O)c(C)ccnc1O 56201,C(=O)(CCCCCC#N)NC(C(=O)NC(C#C)CC(C)(C)C)(C)C1CCC1 56202,Cc1cc2nc(-c3nc(CC(C)C)nn3CC3CCCCC3)ccc2c(=O)n1C 56203,C=CCC(C)(CNC(=O)C(c1ccoc1)NC(c1ccc(CC#N)cc1)=O)CO 56204,Cc1cc2c(cc1C)OC(C(N1CCN(C(=O)CC3(CO)CCC3)C(C)C1)=O)C2 56205,C1(=O)C(C)C(=O)Oc2cc(on2)C(C)O1.C(CC(=O)N(C)C)NC(=O)OC 56206,c1(CC(=O)NCCN(C(=O)CSc2cccs2)CCOC)ccc2c(c1)COC2 56207,CC1CCC(C(N2CCC(CN(C(=O)C(C)(F)F)C3CC3)CC2)=O)CC1C 56208,N1(C(CC2(NC(C3C(C)C3)=O)CCCCC2)=O)C2CCC1CN(C)C2 56209,N1(C(C2(CC)CCN(C(C3CC34CCCC4)=O)C2)=O)CCC(C)(C2CC2)C1 56210,Cc1nc2n(n1)CC(C(=O)NCC1CN(C(=O)CCn3cncn3)CC1O)CC2 56211,c1(OC)cc(C(=O)Nc2ccc(C(=O)Nc3csc(C#N)c3)cn2)ccc1Br 56212,c1(CC)[nH]nc(C(N2CCCC2C2CCN(C(c3cn(C)cn3)=O)C2)=O)c1Br 56213,CN1CC(F)CC1C(=O)NC(Cn1cncn1)C(=O)NCCC1(O)CCC1 56214,S(=O)(=O)(CC(=O)N(CCCNC(=O)Cc1cnn(CC)c1)CCO)NCC 56215,Cc1ccc(C(F)F)cc1C(N1CCC1CNC(c1cccc(C#N)c1)=O)=O 56216,CC1CCC(CNC(=O)CCNS(C)(=O)=O)CN1C(=O)C=CBr 56217,c1(OC)cccc2c(N3CCCC(CC(C)C)C3)ncnc12 56218,c1(N(C(c2cnc(C(C)C)[nH]2)C)C)ccc(C2CC2)cc1 56219,C=C1CCC(C(=O)NCC2(CNC(=O)C(C)OC)CCC2)CC1 56220,C(C(O)CC(=O)NCCC1CN(C(=O)CCc2ncco2)CCO1)N(C)C 56221,C(=O)(CCS(C)(=O)=O)N1CCC(C(=O)N(C2CCOC2=O)C)(OC)C1 56222,C(=O)(CCCC(C)(C)NC(=O)C(C#N)C(C)(C)C)NCC1(F)CCN(C)C1 56223,Cc1ccc(C)c(C(N2CC(CCNC(C3CC(C(C)C)=NO3)=O)C2)=O)c1 56224,c1(N2CCC(C)C2)ncnc2c1ncn2CC1CCCCC1O 56225,CC1(C)COC1C(N1CCCC1CNC(=O)Cc1cc[nH]c1)=O 56226,Cc1scc(C(=O)NCCN(CCCN(C)C)C(=O)CC2CC3CC3C2)c1C 56227,N1(C(CNC(CCC)=O)=O)CCC2CCN(C(=O)Cc3cccc(OC)c3)C2C1 56228,C1(CNC(CC(CC)(C)C)=O)CC2CCC(C1)N2C(C1(COC)C=CCC1)=O 56229,c1(C(N(CCC(C)NC(C2CCC(=O)N2C)=O)C)=O)ccc(N(C)C)cc1 56230,N(C1CCCc2c(Br)cccc21)C(C1N(C(=O)OC(C)(C)C)CC(C)(C)OC1)=O 56231,CC1CCN(C(=O)C(=O)NC2(CCNC(=O)CC3(C)CC3F)CC2)CC1 56232,C(=O)(C1=NOC(C)(C)C1)NCCOCCC(N1CCCC(N(C)CC)C1)=O 56233,c1(C(=O)O)nnc(S(=O)(=O)NC(C2CCCOC2)C(=O)O)s1 56234,C12(CNC(CCCCCC)CC)CNCC(=O)N1CCOC2 56235,c1(CC)cc(NC(=O)COC2(C)CN(C(=O)CNC=O)C2)cc(C)c1 56236,C1(CC(=O)NC(CCNC(CC=CCC)=O)(C)C)CCCC(C)(C)C1 56237,c1(CC)cc(C(C)C)cc(C(F)(F)F)c1.O1NC(=O)CNC(=NC)NC(C)C1 56238,C1(NC(CS(=O)(=O)NC)=O)(CO)CCN(C(=O)Cc2cccc(C)c2C)CC1 56239,c1(NCc2ccn(CC)n2)[nH]c(=NCc2cnn(C3CC3)c2)nc2scnc12 56240,N1(C(C(CC(C)C)(C)O)=O)CC2(C=C(C(=O)NCC3CCSC3)CO2)C1 56241,CCCCC(N)C(=O)N1CCC(O)C(C(N2CCN(C)CC2CCO)=O)C1 56242,N1(C(COC)=O)CC2CCN(C(c3cc(O)cc(O)n3)=O)CCC2C1 56243,C1(NC(C(C)CC2CCCC2)=O)CC12CCN(C(=O)CC1CCCN1C)C2 56244,C1(NC(C(c2cc(C)oc2C)C)=O)CCCCN(C(=O)C(F)(F)c2nccs2)C1 56245,C1(CC=C)(NC(c2oncc2C)=O)CCN(C(=O)CCN(CC(F)(F)F)C)CC1 56246,C1(NC(C2CC(C)(CC)C2)=O)(CO)CCCN(C(=O)C(C)(C)c2nccs2)C1 56247,c1(C(CNC(c2ccon2)=O)NC(C2CN(C)C(=O)C2)=O)ccc(F)cc1F 56248,C(=O)(C(F)(F)CC(C)C)N(C(C)CNC(=O)COc1c(F)cccc1Cl)CC 56249,c1(C(=O)NC(CC)CN(C)C(c2cc(C)cs2)=O)cc(N)c(Cl)c(O)c1 56250,C12CCCCC1NC2=O.C(=O)(C(C(C)C)N(C)C)NCC1N(CCC)CCC1 56251,C1(C(N(C(CF)CF)C)=O)CC1C1CN(C(C2CN3CCC2CC3)=O)C1 56252,C1(CC(=O)NCC(CC)NC(c2nnsc2C(F)F)=O)CC(C)(C)OC(C)(C)C1 56253,N1(C(C2C(C)C2)=O)CCCCC1CNC(=O)CCc1cnn(C)n1 56254,N1(C(Cc2c(C)cnn2C)=O)CC(CNC(C2CCCC23CCC3)=O)C(C)(C)C1 56255,C(=O)(C1=CCCCC1)NC1C(NC(c2c(OC)cc(C)s2)=O)COCC1 56256,C(=O)(CS(=O)(=O)c1ccccc1C)NCC1C2CN(C(C3CC(OC)C3)=O)CC21 56257,c1(N(CCC)C)ccc(C(=O)NCCCN(C(C2CC(CC)CO2)=O)CC)cc1 56258,C1(C(N2CCC(C(C)(C)C)C2)=O)(COC)CCN(C(=O)CN(C)C)C1 56259,O=C(C(O)CC(F)(F)F)NC1CCN(C(=O)C=Cc2cccc(O)c2)C1 56260,Cc1nnc2n1CC(C(=O)OC1CCC1)CC2 56261,O=C(N=S1(=O)CCNC(c2ccccc2)C1)C1CC1CF 56262,c1(C(N2CC3C(CNC(COCCCC)=O)(C3)C2)=O)nccc(Cl)c1C 56263,C(=O)(CCCC1CCCC1)NCC1(CCNC(C(C)N(C(C)=O)C)=O)CC1 56264,N1(C(Cn2ccc(OCCOC)c2)=O)CCC(CO)C12CC2.N1CC(OC)C1=O 56265,N1(C(c2c(C)coc2C)=O)CCN(C(=O)Cn2cc(C#N)cn2)C(C)C1C 56266,C(CC)(C(=O)N1CCC(c2ncco2)C1)N(C(CSCC)=O)C 56267,c1(OC)cc(C(=O)NCC2COC2)c(NC(c2ccccc2C)=O)cn1 56268,c1(C(=O)NCC2(F)CN(C(c3ncc[nH]c3=O)=O)C2)cc([N+](=O)[O-])n[nH]1 56269,C1(C(N2C(CO)CC(OC)C2)=O)CCN(C(=O)C2CCC3(CCC3)O2)O1 56270,C(CC(=O)NC1CC2OCCCC12)(C(C)OC)NC(c1cnc(CC)o1)=O 56271,C1(CNC(c2cc(C(=O)OCC)on2)=O)CC(C(=O)OC)CC(C(F)(F)F)C1 56272,c1(CNC(N2C(C)CSCCC2)=O)c(Br)ccc(Cl)c1F 56273,CC(CC(C)(C)C)C(=O)N1CC2CC(C1)N(C(=O)CNc1ncccn1)C2 56274,Cc1ccn2nc(C(=O)NCCN(C)C(C3CC4CC4C3)=O)nc2n1 56275,Cc1c(C(=O)N(c2nccc(Cl)n2)C)cccc1C(F)(F)F 56276,C1(C(=O)NCC2CC3CCC3C2)CCN(C(=O)Cn2cccc2)C12CC2 56277,c1(OC)ncc(C=CC(=O)NC2CCCN(C(C3CCCN3C)=O)C2C)cn1 56278,c1(CC(=O)OC)cc(C(N2CC3CC2CN3c2ncncc2C#N)=O)cc(Br)c1 56279,C(=O)(CC=C(Cl)Cl)CCN(C)C(CCOC(C1(c2ccccc2)CC1(Cl)Cl)=O)=O 56280,N1(CCN(C(CCC)C)C)CC(C)OC(C)C1 56281,n1(CC)cc(CN(C(=O)CNC(=O)CNC(=O)C(C)CO)C)nn1 56282,CC1CC(CCNC(c2cc(Cl)no2)=O)CCN1C(=O)Cc1ccc(F)nc1 56283,N1(C(c2ccc(CC)[nH]2)=O)CC(NC(C2CC(OC(F)F)C2)=O)CC1C 56284,N1(C(CC(C)CF)=O)C2CCC1CC(NC(=O)CN1CSCCSC1)C2 56285,CC(CCCCNC(=O)CNC(=O)C(F)(F)F)NC(=O)CCn1cccnc1=O 56286,C(=O)(C(C)(C)CNC(C)=O)N1CCC(C(N(CCC)C2CC2)=O)C1 56287,C1(CC(=O)N(C2CCN(C(C(CC)F)=O)CC2)C)CCCC(C)(C)O1 56288,c1(C(C(=O)NCC2CC2)N(CCC)C)cnc(CC)s1 56289,CC1CCCc2cc(C(N3C4CCC3CN(C(=O)Cc3nccn3C)C4)=O)nn21 56290,CC1CC(N(C(C(=O)NCCC2CC2)c2cnc[nH]2)C)CCN1C 56291,C=C(C)CC(C)C(=O)NCC(CC)NC(=O)C(C)(C)C(F)F 56292,N(C(=NCCc1ccccc1F)NCCF)C1(C)CCC1 56293,C(c1cncnc1O)=CC(=O)NCC1CN(C(CCNC(C)=O)=O)C1 56294,CC1CN(C(C2CCC3(CC2)N=N3)=O)CCC1NC(C1SCCCS1)=O 56295,Cc1cc(N)c(C(N2CCC(O)(CCNC(c3ccc(Br)o3)=O)C2)=O)c(F)c1 56296,C1(C(N2CCC(C)(NC(=O)CC3COC(=O)C3)C2)=O)C2Cc3ccccc3C12 56297,C(=O)(CC(C)CC(=O)NC1CN(C(c2cc(C3CC3)no2)=O)C2(CCC2)C1)OC 56298,c1(C(=O)NC(C(C)NC(c2c(C)nc(CCC)s2)=O)C)ccc(OC)nc1Cl 56299,Cc1cn2ccnc(C(=O)NCC(C)(C)NC(=O)C(C)CC(N)=O)c2n1 56300,c1(OC)c(C(=O)NC2CCN(C(c3occc3C)=O)CC2C)cccc1Br 56301,c1(C(=O)NCCCOCCCNC(=O)CC2C=CCC2)cscc1C1CC1 56302,C=CCCCCCCCC(C(=O)NCCC)N1CC2CCCN2CC1C 56303,CC(CCC1CNc2ccccc21)n1cc(Cc2ccccc2)nn1 56304,c1(OC)cnncc1C(=O)NCC(O)CCNC(c1cncnc1)=O 56305,NS(=O)(=O)c1cccc(C(=O)NC2C3CC2CN(C(c2ccc(CO)o2)=O)C3)c1 56306,N12C(CCC1C)C(=O)NC(C)C2=O.c1(C(N2CCCCC2)=O)cnc(Cl)nn1 56307,CCC(CNC(=O)CSC1CCCCO1)(CC)NC(=O)CSC(F)(F)F 56308,C1(CNC(C2CC23CCCC3)=O)CNCCC12CCOCC2 56309,C1(O)(C(C)NC(CC2C(C)CC2)=O)CCN(C(C2(CF)CC2)=O)C1 56310,N1(C(Cc2n(C)nnc2)=O)CC(NC(c2csc(C(N)=O)n2)=O)C2CCCC2C1 56311,c1(CC)nc(C(=O)NC2CC(CNC(=O)C(c3ccccc3)O)C2)c(C)o1 56312,N1(C(CC#C)=O)CC2COCC2(C(N2CCCC2C(C)(C)O)=O)C1 56313,c1(OC)cc(Br)c(C)nc1NC(C1CC(F)CN1Cc1cc(C)n(C)n1)=O 56314,N1(CC(=O)NC(C2(C(=O)OC)CC2)=O)CC(O)CC2(CCNCC2)C1 56315,CCC(CC(C)C)C(=O)NCC1(C(N2CCC(OCCF)C2)=O)CCCCC1 56316,C1(N(C(C(CNC(c2nc(C)sc2)=O)N(C)C)=O)C)COC(C)(C)C1 56317,CCCCN=C(NCCc1ccc2c(c1)OCO2)NC1CCC1(C)C 56318,N1(C(C2N(C(c3c(C)ncc(Cl)c3)=O)CCSC2)=O)Cc2cccc(O)c2C1 56319,N1(C(CCS(N)(=O)=O)=O)CCC2CCN(C(C3(O)COC3)=O)CC12 56320,CC(C)CC(C(=O)N1CCC(O)(CC2CC2N)CC1)ONC(c1ccccc1)=O 56321,C1(CNC(C(CC)SC)=O)CC2(CCN(C(c3ccc(C(C)C)cc3)=O)CC2)C1 56322,C1(NC(COCC=C)=O)CCCN(C(=O)Cc2csc(C3CCS(=O)(=O)C3)n2)C1 56323,C(C(=O)NC1CCCCC1NC(=O)C#CC1CC1)(C(C)C)(C(C)C)NC(C)=O 56324,Cc1ccccc1COCC(N1CC(NC(C2CC3(CC3)CO2)=O)C(O)C1)=O 56325,CCC(C)(CO)CN=c1cc(NC(c2csc(C3CC3)n2)C)nc[nH]1 56326,C1(NC(C(=O)NCC2CCC=CCC2)=O)CCC2C3CCC(C3)C12 56327,CC(C)CCC(F)C(=O)N1CCC(O)(CCNC(C2CCCCCC2)=O)CC1 56328,c1(NC2(COC)CC(c3nnnn3CC(F)F)C2)cc(NS(C)(=O)=O)cc(O)c1 56329,c1(C(=O)NC2CCCC(NC(CN(C)C)=O)C2)ccc(Cl)c(N2CCCC2)n1 56330,c1(C(=O)OC)ccc(F)cc1CCC(N1CC2CCC1C2C(=O)OC)=O 56331,C1(C(=O)NCC(CN(C(C(=O)NCCOCCCC)=O)C)O)C(C2CC2)C1(F)F 56332,C1(C(=O)Nc2ccc(COC)cc2)CCOCCN1C(c1cnn[nH]1)=O 56333,N1(C(=O)COC2CCCOC2)CCC(NC(=O)CSCC2CCCO2)CC1 56334,c1(C(C(N2CC(CNC(CN(CC)CC)=O)OCC2)=O)(C)C)cccc(C#N)c1 56335,N1(C(C(C=C)(C)C)=O)CCC(C(F)(F)F)C(NC(c2nnc(C)cc2O)=O)C1 56336,CCCCC(O)C(C)C(=O)NCC1(C)CCN(C(=O)COCc2nc[nH]n2)CC1 56337,c1(C(N2CC(OCCNC(C3C(C=C)C3)=O)C2)=O)cc(Cl)c(Cl)cc1O 56338,c1(OC)ccc(C2(NC(=O)N(C3CC3)Cc3ccnc(SC)n3)CC2)cc1OC 56339,c1(-n2c(C)ncc2)ccc(CN2CCC(N(CCCn3ccnc3)C)CC2)cc1 56340,N1(C(CCOCCN(C)C)=O)CCN(C(=O)CC2CCC2)C2(CC2)C1 56341,c1(OC)cc(NC(c2c(NC(C34CCCC3C4)=O)cccc2F)=O)nc(OC)n1 56342,C1(C(=O)NCCN(C(=O)COC2CCCOC2)C(C)C)OCC2COCCC12 56343,C1(C(=O)OC)CN(C(=O)C(=O)NCC2(C)CCN(C)CC2)C(C)(C)C1 56344,c1(OC)cc(C2(C(=O)NC3CCC(CNC(=O)CC4CC=CC4)C3)CC2)ccc1C 56345,c1(CC)nc(C)c(C(=O)N(CCCONC(C(C2CC2)OC)=O)C)o1 56346,N1(C(CCCC#C)=O)CCC(NC(C2CCCN(C(C)=O)C2)=O)C1(C)C 56347,CCC(C)(C)C(C(=O)NC1(CNC(c2cscc2C)=O)CCOCC1)OC 56348,C1(C2CC2)(CNC(C=C(CCC)C)=O)CCN(c2cc(C(F)(F)F)nc(C)n2)C1 56349,c1(C(N2CCC(C(=O)O)C2)=O)ccc(F)c(S(=O)(=O)N2CCN(C3CC3)CC2)c1 56350,C1(NC(=O)Nc2ccnc(N3CCOC3=O)c2)CCc2cc(Br)ccc2C1 56351,N1(C(C2=C(C)OCC2)=O)CC2(CCC(NCc3cc(F)cc(Br)c3)C2)C1 56352,C12(NC(c3csc(-c4ccoc4)n3)=O)CC1CN(C(c1cc[nH]c1C1CC1)=O)C2 56353,N1(C(C2N(C(C(C)CC(N)=O)=O)CC3CC32)=O)CC2(C1)NC(=O)NC2=O 56354,Cc1cc(C)cc(C=CC(N2CCCC2CN(C(=O)CCSCC(N)=O)C)=O)c1 56355,N(C1CCNc2ccc(OC)cc21)C(=O)NCC(c1ccc(CC)cc1)(C)C 56356,c1(OC)ccc(OCC(=O)NCC(C23C(CO)(CCC2)C3)NC(=O)C(C)O)cc1 56357,C1(C(N2CCN(Cc3nc(C4CCCCC4)no3)CC2)=O)CC2(CSC2)C1 56358,c1(C(N(C2CCN(C(C(COC)C)=O)C2)C)=O)c[nH]c(=N)c(C)c1 56359,C1(C(=O)NC)C2CC1N(C(c1cnc(Cl)s1)=O)C2.C1(n2cccn2)COC1 56360,C12(NC(c3cc(C)sc3)=O)CCCC1CN(C(c1cc[nH]n1)=O)C2 56361,C1(CNC(CC(C=C)(C)C)=O)CN(C(=O)CCc2nc(C)no2)CC2(CCC2)O1 56362,C1(C(=O)Nc2cccc(C)c2C)(CC)CCN(C(c2sccc2OC)=O)CC1 56363,CCC(CC(=O)N1CC2C(CNC(C3CC4(CCOCC4)C3)=O)C2C1)C(C)C 56364,c1(C(=O)NCC23CC(CO2)N(C(=O)CC=C(Cl)Cl)C3)c(F)ccc(Cl)c1F 56365,C1(NC(C(CC)=CC)=O)CC(C2CCN(C(c3ncnc(C)c3C)=O)C2)C1 56366,C1(OCC(=O)NC(C2CC2C(F)F)=O)CCC(F)(F)CC1.C1CCN1CCCF 56367,C(C)(C)(CN=c1[nH]nc(C#N)s1)SCCNC(c1c(C)cc(Cl)cc1C)=O 56368,C12(NC(C3ON=C(CC)C3)=O)CCCC1CN(C(=O)Cc1csc(C)n1)C2 56369,Cn1cc(CCC(=O)NC(C(N2CCC(c3cnn[nH]3)C2)=O)C2(O)CCC2)cn1 56370,c1(C(C(CC)NC(=O)C(F)(F)Cc2cccc(Br)c2)O)ccccc1F 56371,CC1CC(N(C(=O)C(C)(C)CN(C(=O)Cc2cncnc2)C)C)CC(C)O1 56372,N1(C(C2(c3cccc(OC(F)F)c3)CCC2)=O)CC(NC(=O)C2CC2)CC(O)C1 56373,N1(C(CC(N)Cc2ccc(OC(F)(F)F)cc2)=O)CC2NCCOC2C1 56374,C(=O)(C(C)CC(C)C(C)=O)NC1C(C(=O)NCC2(CC(=O)OC)CC2)CC=CC1 56375,CCCC(CC)C(=O)NCCCNC(=O)C(O)Cc1c(F)cccc1Cl 56376,C(CN=c1[nH]c(=NCC2CN(C)CCN2C)[nH]c2c1COC2)N(CCC)CCC 56377,c1(OC)cc(C(=O)OCC2CCC(CC(F)(F)F)CC2)cc(C#N)c1 56378,c1(C(=O)NCC(c2cccc(Cl)c2Cl)F)cc(Cl)c([N+](=O)[O-])s1 56379,n1(CC)c(NC(=O)CSc2nccc(C(C)C)n2)nc2ccc(Br)cc12 56380,N1(C(c2cc(C)n(C)c2)=O)CC(NC(C2CC3(CCCO3)C2)=O)CCC(O)C1 56381,c1(OC)ccc(C(=O)NCCN(CCC)CC)c(OC(c2cnn(C)c2C)=O)c1 56382,c1(C(N2CCC(F)(C(=O)Nc3ncc(Cl)nc3Br)CC2)=O)cc(Cl)cc(Cl)c1O 56383,C=CCC(C(=O)N(C)CCN(C(=O)C(O)c1ccsc1)C)C(C)(C)C 56384,C(=O)(C(C)(C)S(=O)(=O)C1CC1)NCC(C1N(c2snc(C)n2)CCC1)(C)C 56385,C1(C#CC(=O)NCC(F)CNC(=O)C(c2ccc(O)cc2)(C)C)(CC)CC1 56386,N1(C(c2c(C)nc(O)s2)=O)CCN(C(=O)CCc2cn(C)nn2)CC(C)C1 56387,N1(C(C=COCC)=O)CC(NC(c2cnc(OC(C)C)cn2)=O)CC2(CC2)C1 56388,c1(C(=O)Nc2ccc(F)nc2F)n[nH]c2c1CN(Cc1cc3sccc3s1)CC2 56389,C1(C(NOC(C)C)=O)CCC(NC(=O)COCCF)CC1 56390,Cc1cncc(C(=O)NCCC(C)CCNC(=O)C(F)CC2CCCCC2)c1 56391,CC1=C(Br)CN(C(=O)C(=O)Nc2cccnc2OC(F)(F)F)CC1 56392,c1(C(=O)NCCN(C(=O)C(C)N2CCC2)CC)cc(C(=O)OC)c[nH]1 56393,c1(OC)cc(Cl)c(-c2cn(CC3CCCN3C(=O)Cc3cnns3)nn2)cc1Cl 56394,c1(C(N2CC3C(C(=O)Nc4c(C)cc(Cl)nc4)C3C2)=O)ccc(F)c(C#N)c1 56395,c1(SC)cc(C(=O)NCC2CC(F)(CNC(=O)Cc3csnn3)C2)c(C)o1 56396,c1(CCN2C3CCN(C(=O)OC(C)(C)C)C3CCC2)ccc2cc(O)ccc2c1 56397,C1(NC(CC2N(C(C(C)SC(C)C)=O)CC(O)C2)=O)CCC(C)(C)CC1 56398,Cc1cc(NC(=O)CSCCNC(C2CC3(C2)CC32CC2)=O)c(F)cc1F 56399,C(CC(C(=O)N(C)CCO)NC(=O)CSCCOC)SC 56400,C(=O)(CS(=O)(=O)CC(=O)OC)NC1C(NC(C(COC)C)=O)CCC1 56401,CC1CC(C(=O)NCC2(F)CN(C(c3cc(O)cc(O)n3)=O)C2)Cc2nn[nH]c21 56402,C1(C(=O)NC2CC(CO)C23CCC3)(CC)CCCN(C(=O)C2=COCCC2)C1 56403,N1(C(c2cc(C)nc(O)n2)=O)CC2(CCCN(C(c3ccc(CF)cc3)=O)C2)C1 56404,C1(C)(NC(c2ccc(C(C)C)nc2)=O)CCN(C(C2CCC(F)C2)=O)CC1 56405,CC1CC(=O)NC(C(=O)NC(C2CC2C(=O)NCC=C2CCSCC2)C)C1 56406,C(C(C)(C)C#CC(=O)NC1C=CCCC1)NC(Cn1c(C)ccc1C)=O 56407,Cc1cnc(C(=O)NC(C2(O)CN(C(=O)C3=CCCOC3)C2)C)cc1C 56408,C1(NC(CCCCSC)=O)CCN(C(=O)CCOCC(C)(C)C)CCC1CO 56409,c1(C(=O)NC2C(NC(C(=Cc3cccs3)C)=O)CCC2)cc(Cl)ccn1 56410,N1(C(c2c(C)cc(CNC(CCSC)=O)o2)=O)CCC2(C1)CC2(F)F 56411,N1(C(c2c(CC)[nH]cc2)=O)CCN(C(=O)C(C)NC(C)=O)CC1C(F)F 56412,Cc1cncc(C)c1C(N1CCOC(CCNC(C2CCC(C)(C)OC2)=O)C1)=O 56413,CC1CCC(C(=O)NCCCCCF)N1C(c1ccc(C2CC2)cc1)=O 56414,C1(NC(CCC#CC)=O)CCN(C(=O)Cc2c(C)noc2Cl)CC1C 56415,C1(O)(CCNC(C2C(C(C)(C)C)C2)=O)CN(C(C2CC(=C3CCC3)C2)=O)C1 56416,C1(OC)CCC(C(N2CC(N(C)C(c3cnn(C(C)C)c3F)=O)C(O)C2)=O)CC1 56417,c1(OC)cc(CN(C(c2csc(Br)n2)C(=O)NCCC2CC2)C)c(OC)cc1C 56418,CCC(C)(CO)C(=O)N1CC2(CCN2C)C1 56419,CCCCCC(F)C(=O)NC1CCSC12CN(C(c1cnc(O)o1)=O)C2 56420,C1(NC(CCC=CC)=O)C(C)CCN(C(=O)CC)C1C 56421,C1(CCC(=O)NCCC(C)(C)F)CCCCN(C(=O)C=CC2CCOCC2)C1 56422,CC1CN(C(=O)Cc2ccn(C)n2)CC1(C)CNC(C1CC(F)C(=O)N1)=O 56423,C(CC(C)C(=O)N(C(C)C(=O)N(C1CC(C)(C)C1)C)C1CC1)=CCC 56424,CC(O)CC(C)(C)CNC(C1(F)CCN(C(C2(C(F)(F)F)CC2)=O)C1)=O 56425,c1(C(=O)NCC(CC)N(C)C(c2csc(F)c2)=O)ncc2[nH]ncc2n1 56426,Cc1ncccc1NC(=O)C(C)CN(C(=O)C(C)O)C 56427,C(C(=O)NC1CCCC1(F)F)(C(C)OC)NC(C(CC)=CCCC)=O 56428,N1(C(C2(CCOC)CCC2)=O)CCC(NCCCC2CCOC2)C(C)C1 56429,C=CC1(CC(N2CCCC(CO)(NC(=O)CN3CCCC3C)C2)=O)CCCCC1 56430,c1(C(=O)NCC2N(C(C(CC#C)C)=O)CCC(C)C2)ccc2nc[nH]c2c1F 56431,C(=O)(C(CC)CC(F)(F)F)N1CCC(CNC(c2cc(CC)on2)=O)C12CC2 56432,c1(C(N(C2CCN(C(c3c(CCC)nns3)=O)CC2)CC)=O)cc(C)ccc1F 56433,c1(N2CCC(NC(C3C(C)=C3)=O)C(C)C2)ncc(C#N)cc1Br 56434,C(=O)(C1=C(C#N)CCC1)N1CC(NC(c2ccc(-c3nc(C)on3)cc2)=O)C1 56435,c1(OC)cccc(CNC2C(C(=O)C(F)(F)CSC)CC2O)c1 56436,N1(C(c2cc(C)oc2)=O)CCN(C(c2ncc3[nH]ncc3n2)=O)CC2(CC2)C1 56437,CC1CC(C(N2CCC(O)(CN(C(=O)C3=COCCO3)C)CC2)=O)CC(C)O1 56438,c1(CCC(=O)N(CCCNC(C2CC3(F)CC2C3)=O)C)ccc2c(c1)CCO2 56439,C1(C)(CNC(C(c2cccs2)NC(c2ccn(C)c2)=O)=O)CC2CCC1C2 56440,Cc1ccnc(CNC(=O)CC2CN(C(=O)OC(C)(C)C)CC2C)n1 56441,C=CC(C)(C)CC(=O)NCC1CN(C(=O)C=CC2CCC2)CC1O 56442,c1(NC(C(C)(C)C)=O)ccc(NC2(c3cccc(Br)n3)CCC2)cc1 56443,C1(CNC(CCCN(C(C)=O)C)=O)CCCCN(C(c2cc(C(F)F)no2)=O)C1 56444,C1(F)(C(=O)OCC)CN(C(c2cn[nH]c2C(C)C)=O)CC12CNC2 56445,N1(C(CN(C(=O)COCC(C)(C)C)CCOC)=O)CCC(CO)(CO)C1 56446,c1(C(=O)NC2(C)CCN(C(C(=O)N(C)C)=O)CC2)cccc2c1OC(C)(C)CC2 56447,Cc1csc2c(C(N3CCCCC3CNC(=O)CC34CCCC3C4)=O)cccc12 56448,C(=O)(C(C)CC(C)(C)C)NCC(CC)N(C(=O)CSC(F)F)C 56449,c1(C(N2CCCC(N(C(c3nc(C)c(C)s3)=O)CC)C2)=O)nc(C)ccc1F 56450,C(=O)(C(F)CC(C)C)NC1(CCOC)CCN(C(CC=C=C)=O)C1 56451,C1(C)(CC(=O)NCC(C)Cn2ccnc2)CCN(C(=O)CC2CC(C)(C)C2)C1 56452,c1(C(=O)NCCCC(C)NC(c2cc(C(=O)OC)sn2)=O)ccc(=O)oc1 56453,N1(C(C(C)OCC)=O)CC2(CCCC(CNC(c3nn(C)cc3[N+](=O)[O-])=O)O2)C1 56454,C(N=c1[nH]c(=NCC(=O)N2CCCO2)c2c(F)cccc2[nH]1)c1scc(CC)n1 56455,Cc1cc(C=CC(=O)NCC2(O)CCCN(C(c3cnnn3C)=O)C2)ccc1F 56456,N(C(=NCc1nccs1)NCC(C1CCOCC1)O)C(COCC)C 56457,C=C(CNC(=O)Cc1ccsc1)CCNC(C1CCN1C(C)=O)=O 56458,C=C(C)C(C)(C)C(=O)NC1CCC(C)(CNC(=O)CNC(C)=O)CC1 56459,C(c1ccccc1F)=CCC(=O)NC1(CNC(=O)Cc2cc[nH]c2)CCOCC1 56460,c1(OC)cc(CNC(C2CCCC2NC(=O)CCC2CC2)=O)cc2c1OCO2 56461,c1(C(=O)NC2C(CNC(CC(=O)N(C)C)=O)CCC2)cc2cc(Cl)c(Cl)cc2[nH]1 56462,C1(NC(CC(C)(C)C)=O)CCN(C(=O)COc2ccccc2Cl)CC(O)C1 56463,C1(N(C(C(C)C2CC2)=O)C)CN(C(=O)Cc2c(F)cncc2Cl)CCC1O 56464,c1(OC)cc(CN2CCCC2CNC(c2cc([N+](=O)[O-])cs2)=O)c(OC)cc1C 56465,c1(C(=O)NCc2ccc(OCCC)cc2)nc2ccc(-c3cnn(C)c3)cn2n1 56466,c1(N(C(c2ccco2)=O)CC)ccccc1C 56467,C(=O)(CCCCCC(C)(C)C)N1C(CNC(=O)C=C(C)C2CC2)CC(COC)C1 56468,Cc1cnsc1C(=O)NC1(CCC(=O)NCC2CCC(C3CC3)O2)CCCC1 56469,N1(C(CCCC2(NC(C=C(C)C)=O)CCC2)=O)CC(S(C)(=O)=O)C1 56470,c1(C(N2CC=CC(NC(C(C=C=C)C)=O)C2)=O)cc([N+](=O)[O-])n[nH]1 56471,N1(C2CCN(C(CCNC(=O)OC)=O)C2)CCN(C(C2CCCSC2)=O)CC1 56472,N1(C(c2cncc(SC)c2)C(=O)NC(C(=O)OC)C)CCC(O)C2CCCCC12 56473,C1(CC)CN(C(=O)COCC2CC2)CCC1NC(C1CC(O)(C#N)C1)=O 56474,CCCC(C(=O)N(CCNC(=O)C(c1ccccc1)F)CCOCC)NC(N)=O 56475,c1(NC(c2ccc(CCC(N3CC(F)C(F)C3)=O)[nH]2)=O)cnnc(Cl)c1 56476,C1(NC(CN(C)Cc2nnc(C)n2C)=O)CC2CC1N(C(C1CC=CCC1)=O)C2 56477,N1(C(CC2C(C)(C)CCCO2)=O)CC2CC(C1)CN(C(C1C(F)(F)C13CC3)=O)C2 56478,Cc1ccccc1N=c1[nH]c(CN2CCCS(=N)(=O)CC2)nc(=N)[nH]1 56479,c1(NC(c2ccc(-c3cn(CCOC)nn3)cc2)=O)nc(C)c(C)c(C)c1C#N 56480,Cc1nc2sccn2c1C(=O)NC1(C2CCCN2C(C2COCCO2)=O)CC1 56481,CC1(C(=O)NCC(c2ccc(O)c(O)c2)O)CCCN(CCN2CCCCC2)C1 56482,c1(C(=O)NC2C(NC(C(COCC)(C)C)=O)CCC2)ccc(P(C)(C)=O)nc1 56483,c1(C(C2CC2)OC)nc(C2CCCc3ncnn32)n(-c2ccc(C(C)C)cc2)n1 56484,c1(C(N(C2CCCN(C(=O)C(F)=CCCF)C2)CC)=O)cnc(C2CC2)nc1O 56485,CCN=c1ccc(C(=O)NC2CN(C(c3ccc4cnoc4c3)=O)CC2C)c[nH]1 56486,c1(CCC)nccn1CC(=O)NCCN(CCC)C(C1CC(n2cnnc2)C1)=O 56487,C1(CC=C)(C(=O)N(C(C)C(C)SC)C)CCN(C(=O)C(CC2CCC2)OC)C1 56488,N1(C(c2c(SCC)nccn2)=O)CCN(C(=O)C2=CCCC2)C(C(C)C)C1 56489,C1(C(=O)NCCC(C)NC(c2c(C)onc2CO)=O)CCCCN1S(N)(=O)=O 56490,C1(NC(Cc2cc(CC)nn2C)=O)CC(O)CN(C(=O)CCC2(C)CC2)C1 56491,c1(C(=O)NC(CNC(CN(CCC)C)=O)C(C)C)cc(C)c(C)c(S(N)(=O)=O)c1 56492,c1(OCC(=O)NC(CN(C(c2cnc(C(=O)OC)s2)=O)C)C)ccc(F)cn1 56493,CCC(C)C(O)C(C)C(=O)NCC(COC)NC(=O)C(O)CSC1CC1 56494,CC1C(NC(=O)C=Cc2nccs2)CCCN1C(=O)CC(C)c1ccccc1 56495,Cn1ncc(C(N2CCCC2CNC(c2cnn(C3CCC3)c2)=O)=O)n1 56496,c1(OC)c(Cl)ccc(C(=O)NC2(C)CN(C(c3cc(N(C)C)ccn3)=O)C2)c1N 56497,C1(C(N2CCCCC2C2CNC2)=O)CC(F)(F)CCO1 56498,N1(C(C(C(=O)OCC)F)=O)CCC(NC(c2ccc(CC)cc2F)=O)C12CC2 56499,C(CCN=c1[nH]c(=NC(C)c2ncc3ccccn23)[nH]c2c1CSC2)OC 56500,C(C)(CC(C)NC(=O)CNC(c1cscn1)=O)NC(C1(CCOC)CCC1)=O 56501,N1(C(CN(C(C)=O)C)=O)CC(O)CC1CNC(=O)C(CO)c1ccccc1 56502,c1(OC(F)F)ccc(-c2ncn(C3CCC3)n2)cc1.C1(C2CC2)CCCO1 56503,C1(NC(c2cc(C)cc(F)c2)=O)CCC(O)CN(C(=O)COCC(F)(F)F)C1 56504,N1(C(c2cc(C3(C)CC3)n[nH]2)=O)CCC(CNC(=O)Cc2cnc[nH]2)C(O)C1 56505,N1(C(c2csc(C)c2C)=O)C(C)CC2CN(C(=O)CCC3(C)CC3(F)F)CC12 56506,Cc1ccc2oc(C(=O)NC3(C)CC(C(=O)NC4CCCCC4)C3)cc2n1 56507,CCC(CC)(CC)C(=O)N1CCN(C(=O)Cc2nc(C(C)C)c(C)s2)C(C)C1 56508,N1(C(c2nc(COC)oc2)=O)CCN(C)C(CNC(c2cc3ccsc3[nH]2)=O)C1 56509,C(=O)(CCCN=[N+]=[N-])NCC(C)CNC(c1cc(C2CCCN2C)[nH]n1)=O 56510,C(N=c1[nH]c2cc(Cl)c(S(=O)(=O)NCC(Cl)(Cl)Cl)cc2s1)C1C(C)OCC1 56511,C1(NC(c2c(CC)ncs2)=O)COC2(C1)CN(C(C1(C)CCC(C)CC1)=O)C2 56512,C1(F)(CNC(C2CCC(=C)CC2)=O)CCCN(C(C2(F)CC=CCC2)=O)CC1 56513,N1(C(c2cccc(C)c2Br)=O)CC(NC(C2(O)CCC2)=O)CC12CCCC2 56514,c1(Cc2ccc(C(N3CCCC3CF)C(=O)NCC(F)F)cn2)ccc(F)cc1 56515,C1(C(=O)NCC(CC)N2CCCC2)CCCCN1C(C1CC(F)CN1C)=O 56516,C1(CNC(C2CC3CCC2O3)=O)CN(C(=O)CSc2ccccc2O)CC1(F)F 56517,CC1(NC(=O)CCNC(=O)C=CCl)CCCN(C(C2CCS(=O)(=O)C2)=O)C1 56518,N1(C(C(C)SC(C)C)=O)CCCCC(C(=O)NCC2CCCOC2(C)C)C1 56519,c1(C(C)C(=O)NCC(C)N(C(=O)CCOCCOC)C)ccc(F)cc1 56520,N1(C(=O)OC(C)(C)C)CCC2CCN(Cc3ccccc3)C2C1 56521,CCS(=O)(=O)CC(=O)N(C)CCn1cc(-c2ccc(Cl)c(F)c2)nn1 56522,c1(CC(N2CC(CC(C)NC(c3occc3F)=O)C2)=O)ccc(Br)cc1F 56523,C12(CCCCC1)CCC(=O)N2Cc1c(CCC)c[nH]c1.c1(C(=O)NC)ccco1 56524,c1(C(=O)NC2C(NC(C=CCC)=O)CC2)cc2ccc(Cl)cc2c(=O)o1 56525,Cc1c(C(=O)OCC(c2cccc(Cl)c2)=O)cc(Br)cc1[N+](=O)[O-] 56526,C(=O)(CC(C)(C)Cc1ccc(Cl)cc1)NC(CC)(C)CNC(c1cccnn1)=O 56527,n1(CCCCSC)nnnc1C(c1cccn1C1CC1)NCCC1(C)CC1 56528,c1(C(N2CCCC(CCC(=O)NCCCNC(=O)OC)C2)=O)ccc(C)c(O)n1 56529,C12(C(=O)OC)CC1CN(C(=O)C(CNC(=O)C(C(C)C)N(C)C)OC)C2 56530,CCCC(C(=O)NC(C(=O)Nc1cnn(C)n1)C1CCCC1)NC(N)=O 56531,c1(N2CCOCC(NC(CC(C(F)(F)F)OC)=O)C2)nc(Cl)nc2c1ncn2C 56532,C#CC1CN(C(=O)Cc2ncc(F)cc2F)CCN1C(C1CCC=CCCC1)=O 56533,c1(-c2cn(CCN(C(C=C(CC)CC)=O)C)nn2)c(F)cccc1F 56534,C1(NC(Cc2nc(C)sc2C)=O)CC2(NC(=O)C(C)n3ccnc3)COC1C2 56535,Cc1cc(=NCCCC(C)(C)NC(c2ncc(F)cn2)=O)[nH]c(C(F)(F)F)n1 56536,C1(C(C)C)CCN(C(=O)C(C#N)C2CC2)CC1.C(=O)(CC(C1CC1)C1CC1)N 56537,C1(C(=O)NCCCc2nc[nH]n2)CC2C=CC1N(C(=O)CC1CCC=CCC1)C2 56538,C(=O)(C(F)C1=CCCCC1)N1C(CN(C(COCCSC)=O)C)CCC1 56539,c1(C(=O)NC2C(NC(C(Br)=C(C)C)=O)CC2)cc2ncccc2o1 56540,N1(C(c2ccnc(C)n2)=O)CC2CCCCN2CC1CNC(c1oncc1C)=O 56541,N1(C(C(C=C)O)=O)CC2CCC1C1CN(C(c3c(F)cc(F)c(F)c3F)=O)CC21 56542,C1(OC)COCCC1(c1nnnn1C1CCC1)NCCC(=O)Nc1ccccc1 56543,c1(C(=O)NC(C)CCCNC(=O)CC2CCCS2(=O)=O)ncccc1C#N 56544,O=C(C(F)CC1CC1)NC1CCCC1NC(c1cnn(CC2CC2)c1)=O 56545,C(=O)(C(C)C(C)CC)N1CCC(Cc2ccc(OCC#C)cc2)C1C 56546,c1(C(=O)OC)ccc(CN(C)C(C2CCCN(C(=O)OC(C)(C)C)C2)=O)cc1Cl 56547,N1(C(c2ccc(OCC)cc2)=O)CCN(C(C2(C)CC2C)=O)CC1c1cn[nH]c1 56548,CCC(c1ccc(C)cc1)=CC(=O)NC(C)CNC(c1n[nH]cc1OC)=O 56549,c1(C(N(C)CCOCCN(C)C(C2(C)CC2F)=O)=O)ccc2c(c1)OCC2 56550,N1(C(C2CCCC(OC)C2)=O)CC2(CCN(C(c3ccc4c(c3)NCC4)=O)C2)C1 56551,C(=O)(CCC(=O)NC(C)CC1CCN(C(C)C)CC1)NC.C1(C)(C)CC(=O)N1 56552,CC1(CNC(C2CC2c2cccc(O)c2)=O)CCCN1C(c1ccc(Cl)[nH]1)=O 56553,C1(SC)CN(C(c2c(C)nsc2C)=O)CC1NC(=O)CCc1cscn1 56554,c1(SCC)ccccc1-n1nc(C(C)OC)nc1-c1cccc(C2CCOC2)c1 56555,c1(C(c2nnnn2CC(F)F)NCCCc2n(C)ncc2)snc(OC)c1Br 56556,N1(C(CC(CC)(C)C)=O)CCC2(CCCN2C(c2sccc2C)=O)C1 56557,C1(C(=O)NC2CCCC2NC(C2(CO)COC2)=O)CC12CC(F)(F)C2 56558,CCCCC(C(=O)NCC1(F)CCN(C(=O)C(O)(C2CC2)C2CC2)C1)C(C)C 56559,N1(C(C(F)=CC)=O)CCC(C2CCCN(C(c3n[nH]c(CC)c3Cl)=O)C2)C1 56560,C12(NC(=O)CC3CC3)CC1CN(C(C1CCCOC1c1cc[nH]n1)=O)C2 56561,C1(CNC(C2C(CC)OCC2)=O)COCCN(C(c2cnsn2)=O)C1 56562,c1(C(=O)OC)cc(Cl)c(OC)cc1CN1CCCC(CS(C)(=O)=O)C1 56563,C1(OC)CC2(C1)CC(C(=O)NCC1CC3CC3N1C(=O)CCCC(N)=O)C2 56564,N1(C(C2CC2C2CC2)=O)CC2(CNC(C34CCCC(O)(CC3)C4)=O)CC1CCO2 56565,Cc1nc(C(C)C)oc1C(=O)NCC1CCN1C(C1(c2ccccc2)CC1C)=O 56566,C1(NC(CC(CC)O)=O)CC2CCC(C1)N2C(=O)C(c1ccc(F)cc1F)C 56567,C(C#N)(c1ccccc1)=C1CCCN(Cc2cnc(C3C(C)C3)s2)C1 56568,C(=O)(C(=O)N=c1ccn(C2CC2(F)F)[nH]1)N1C(c2n(C)cnc2)CCC1 56569,C(CNC(=O)CN=[N+]=[N-])(CC(=O)NC1C(C)CCC1C)OC 56570,C1(NC(C(C)NC(=O)NC)=O)CCN(C(c2c(C)cc[nH]c2=N)=O)CCC1(F)F 56571,c1(C(N2CC(C(C)(C)O)(CNC(C3C(OCC)CC3)=O)C2)=O)nn(CC)nc1C 56572,c1(OC)cc(C(=O)NCC(COC)NC(C2(C)CCCCC2C)=O)cnc1C 56573,N1(C(C2C(C)(CC)C2)=O)CC2(C(=O)Nc3cn(C)nc3C#N)CCC1CC2 56574,c1(CN(c2ccc(OC)cc2)C)ccc(C)nc1O 56575,N1(C(=O)CCc2nc(O)n[nH]2)CC2CC(N=c3[nH]nc(C(F)(F)F)s3)CC1C2 56576,N1(C(c2cn(C)c(=O)cn2)=O)CC2CCN(C(=O)CC=C(Cl)Cl)CCC2C1 56577,CC1NC(=O)CCC1N=c1cc[nH]cc1S(=O)(=O)NCCCC(N)=O 56578,c1(CC(=O)NCC2=CCN(CCOCC3CC3)CC2)cccc2cc[nH]c12 56579,C1(CNC(N)=O)CCN(C(=NCCCc2nccs2)NCc2ccco2)C1 56580,N1(C(CCc2cc(OC)no2)=O)CC(NC(C2CC2CC(C)(C)C)=O)C2(CC2)C1 56581,c1(C(N2CC(NC(C3CC4CSCC(C3)C4)=O)C2)=O)ncc2[nH]ncc2n1 56582,N1(C(C(C)=C(C)C)=O)CCC(NC(C2(C)CC2(F)F)=O)C(C)C1 56583,C1(OC)CN(C(C2CC3(CCC3)C2)=O)C(C)(CNC(c2ccc(F)cc2Cl)=O)C1 56584,N1(C(c2c(C)cns2)=O)CC(NC(=O)Cn2cc(C#N)cn2)C(C(F)F)C1 56585,CC1CCC(Cl)=C(C(=O)Nc2nc(-c3ccc(Br)s3)cs2)C1 56586,C(=O)(C1CCCc2nncn21)NCC1CCN(C(C2C(C(=C)C)OCC2)=O)CC1 56587,N1(C(C(C(C)C)OC)=O)CCC(CCNC(=O)C(C)(C)O)C(F)(F)CC1 56588,c1(CN2CCN(C(c3cn(C)nc3CC)C(=O)NCC)CC2)ccc(F)c(C)c1 56589,N1(C(c2cc(C)sc2N)=O)CCC2(CC2)CC1C(=O)NCC1CCOCC1(C)C 56590,CC(C)C(O)CC(=O)N1CC(F)CC1CC(=O)Nc1ccc(Cl)nc1 56591,Cc1ccc(C(=O)NCC(=C2CN(C(c3ncccc3Cl)=O)C2)F)cn1 56592,C1(CC(N2C(COC)CCC2)=O)(NC(=O)Cn2nccn2)CCCCC1 56593,c1(NCCC(N2C(C)CC(CNC(=O)C(F)(F)F)C2)=O)ccccc1[N+](=O)[O-] 56594,C(c1cnc[nH]1)=CC(=O)NCC1(CNC(c2ncoc2C(F)(F)F)=O)CCCC1 56595,c1(C(N(C)CC2CCN(C(CCCCCC)=O)C2)=O)ccc2cccnc2c1 56596,c1(OC)ccc(C2CC2C(=O)NC2(C)CC(NC(=O)Cc3ccc(C)s3)C2)cc1 56597,CN1CCC(C(N2CCCC2CCC(=O)N(C2COC(C)(C)C2)C)=O)C1=O 56598,CC(C)(F)CCC(=O)NCC1CCC(CNC(=O)CC2COC(C)(C)CO2)CC1 56599,O=C1NCc2cc(C(=O)NCCNC(c3ccccc3Br)=O)ccc2N1 56600,C1(NC(C2OCCN(CC)C2)=O)(CC)CCN(C(C2(C(N)=O)CCC2)=O)CC1 56601,C1(NC(c2ccccc2CO)=O)CN(C(=O)CC2CCNC2=O)CC(F)(F)C1 56602,C1(C(N2CC(N3CCC3)C2)=O)CCC(O)CN1C(C1CC2(CSC2)C1)=O 56603,N1(C(C(C)OC)=O)CC2CCC(C1)C(NC(c1cccc(OC(C)C)c1)=O)C2 56604,N1(C(CCc2nc(C)c(C)[nH]2)=O)CCCC2CN(C(c3cnccn3)=O)CCC12 56605,C1(C2CCN(C(=O)CCc3nc(-c4ccco4)no3)C2)(NC(CC=C=C)=O)CC1 56606,CC1(C)CN(C(c2ccc(=N)[nH]c2)=O)CCC1NC(c1ccc(C(N)=O)cn1)=O 56607,N1(C(c2ncc(C(F)F)cc2F)=O)CC=C(c2cccc(Cl)c2)CC1 56608,N1(c2nccc(OCC)n2)CCC(C)C(NC(C2CC(C)CO2)=O)C1C 56609,Cc1ccc(C2=CCC3(CN(C(C(=O)NCCCF)C4CC4(Br)Br)C3)CC2)cc1 56610,Cc1[nH]c2ncccc2c1C(=O)NC1CN(C(c2nn[nH]c2Cl)=O)C(C)(C)C1 56611,C=CC1(C(N2CCOC(C#N)C2)=O)CCN(C(c2cc(CC)no2)=O)CC1 56612,C(=O)(C1=C(C)S(=O)(=O)CC1)NCCCNC(c1c(CC)ncc(Br)c1)=O 56613,C(=O)(C(C)(Cc1ccncc1)N1CCN(C)CC1)OC 56614,N1(C(C)=O)CCCC2C1CCN2N1CSCC1C#N 56615,C(CCCCC(=O)N1CCCC(NC(=O)COCC2(F)CC2)C1C)SC 56616,c1(CC)ccc(C)cc1C(=O)NC1CN(C(c2cc(Cl)n(C)n2)=O)CC1C 56617,N1(C(Cc2c(C)noc2)=O)CCC2CN(C(c3cccc(=O)n3C)=O)CCC2C1 56618,C#Cc1cc(N(C(=O)CC2CCN2C(=O)C(=CC2CCCC2)C)C)ccc1C 56619,C(CCCOC)(C(=O)NCCC(C)N(C)CC)NC(c1c(CC)cno1)=O 56620,c1(NC(=O)CNC(=O)NCCC2CCCN2Cc2cccnc2)ccc(F)cc1 56621,c1(C(N2CCC(C(C)(C)NC(C(C)O)=O)CC2)=O)cc2occc2s1 56622,c1(C2C(C(=O)NCC3C(CNC(C(N)=O)=O)C3)C2)ccc(F)c(F)c1 56623,c1(CC)nnsc1C(=O)NCC(C)(O)CNC(=O)CCC1CCCOC1 56624,C(=O)(C(C)(O)CC(F)F)NCC(CNC(CCn1c(C)nc(C)n1)=O)(C)C 56625,c1(C(C(N2CCC(NC(C(C#N)C3CC3)=O)(CO)C2)=O)=O)ccc(F)cc1F 56626,O(NC(=O)C(CCOC)NC(=O)C(C)COC)C(C=C)C 56627,CC(C)(CC(=O)NCC(C)(C)NC(=O)Cn1nnc(=N)[nH]1)CC(F)F 56628,c1(CC(C)C)ccc(C=CC(=O)NCC2CC(CNC(=O)CO)CO2)cc1 56629,Cc1ccc(-n2cc(C(C)N(C)C(C3CCN(C)C3)=O)nn2)c(Br)c1 56630,C(=O)(C(O)CC(F)(F)F)N1CC(CC(C)NC(=O)C(C)(C)C(F)(F)F)C1 56631,C1(NC(c2cc(CO)[nH]n2)=O)C2CCCC1CC(NC(C1(Cl)CC1(F)F)=O)C2 56632,c1(NC(C2(CC)CN(C(=O)CN3CCCC3)C2)=O)cnc(C)c(C)c1C 56633,C=CCCCCC(=O)NCc1csc(CCC)n1 56634,C1(C(N2CC3CC(NC(=O)CCc4cnn[nH]4)C2C3)=O)(CC)CCC(F)(F)CC1 56635,C(=O)(N=c1[nH]c(S(C)(=O)=O)ncc1Br)c1c(Cl)ncc(-c2c(C)cccc2)c1 56636,N1(C(Cc2c(C)cco2)=O)CCc2sccc2C1CNC(=O)C(Cl)=CCl 56637,N1(c2nccc(OCC)n2)CC2(C)CN(C(c3ccncc3)=O)CC2(C)C1 56638,CC1CC(C(=O)NCC2CC(C(=O)NC3(C)CC=CC3)C2)CCS1 56639,C1(N=[N+]=[N-])(C(N(CC(CCCC)CC)C)=O)CCN(C(=O)C2=CC(C)(CC)C2)C1 56640,C1(C(=O)NCC(N2CCOC2=O)C)(CC)CCCN1C(=O)COCC 56641,C1(NC(CCc2ncc(C)[nH]2)=O)(CO)CCN(C(c2occc2Br)=O)CC1 56642,S(=O)(=O)(c1cccc(C(F)(F)F)c1)CCN1CC2N(C(C#C)=O)C2C1 56643,c1(C(=O)O)ccc2c(c1)CCC2NC(c1nc(F)ccc1Cl)=O 56644,C1(COC)(NC(=O)C(C)CC(N)=O)CCCN(C(=O)Cc2cccnc2O)C1 56645,c1(CC)ccc(C(c2nnnn2C2COC2)Nc2ccc(C)nc2)c(C)c1 56646,N1(C(CC=C)=O)CCC(CNC(c2nccc(SC)n2)=O)C(C)C1 56647,Cc1nc(C(N2CC(NC(c3cn(C)c(=O)n3C)=O)C3CC23)=O)c(C)n1C1CC1 56648,C(=O)(NN1CCCC1C(=O)NCCCN(C)C)c1c(C)ncs1 56649,CC(C)CC(C(=O)NC(C1CCCC1)C)ONC(c1ccc(N)cn1)=O 56650,C(=O)(C(O)CC(C)C)N1C(CCNC(c2c(OC)noc2C)=O)CSCC1 56651,c1(C(=O)NC2C(NC(C3(CCOC)CC3)=O)CCOC2)cnc(O)c(Br)c1 56652,N1(C(CCOCC(C)C)=O)CC2(CCC(NC(=O)C(=O)NCC(F)(F)F)CC2)C1 56653,c1(C(=O)NCC2C(NC(CCOC)=O)CC2)ccc(CN2CCCCC2=O)cc1 56654,c1(NC)c(C(N2CCN(C)C(CF)C2)=O)sc2nccnc12 56655,C1(C2(O)CCOCC2)(C(N2CCC(NC(C3C(=C)C3)=O)C2(C)C)=O)CC1 56656,C=CCC(CC(=O)OCC)OCC.c12ccc(cc1)ONCCCNC2=O 56657,N1(C(c2ccc(SCCCC)cc2)=O)CCC2C(NC(=O)CC)CC12 56658,C1(C(=O)NCC(O)C(=O)NC2CC(CO)C2)CCC(O)CC1 56659,CN1CCN(C(=O)CO)CC1COCC(=O)NCC1CCCO1.c1ncnn1C 56660,Cc1nc(C2CC2)ncc1C(N1CCOC(C2(O)CC2)C1)=O 56661,C(=O)(C(CC(N)=O)NC(=O)CCn1cncn1)N(C(CC(C)C)C)C 56662,C1(c2nnnn2C2CC2)(NC2(CC=C)CC2)CCCN(C)C1 56663,C(=O)(C1=CCCN(C(C2CCN(C(c3ccc[n+]([O-])c3)=O)CC2)=O)C1)OC 56664,c1(CONC(c2ccc(CNC(CC(C)(C)O)=O)o2)=O)ccc2c(c1)CC2 56665,c1(C(=O)NC2CC(O)(CNC(C3C(C)C3)=O)C2)cnc2[nH]nnc2c1 56666,CC1(CC(N2CCC(OCC3CC3)C2)=O)CN(C(=O)CCN2CCC2)C1 56667,c1(C(N2CCN(C(C(CC)C)=O)C(c3ccccn3)C2)=O)ccn2cncc2c1 56668,c1(CCC(=O)N(CCNC(=O)CC(C)C)CC)cccc(C(F)(F)F)c1 56669,N1(C(C)C)CCN(C(C23CC(CN2C(=O)C(F)(F)CO)C3)=O)CC1 56670,c1(C(=O)O)ccc2ncc(Sc3n[nH]c(C=Cc4ccccn4)n3)n2c1 56671,C1(NC(C(C)Cc2cccnc2)=O)COCCN(C(c2cc(F)ccc2N)=O)C1 56672,c1(C(=O)NCC(CNC(C2C(C(C)(C)O)C2)=O)O)ccc2ccoc2c1 56673,C(=O)(C1=NOC(C)(C)C1)N1CCC(C(C)NC(=O)C=CC(N)=O)C1 56674,c1(NC2C(Cn3cc(-c4n(CC)ncc4)nn3)CCC2)ncccc1OC 56675,C(=O)(C(O)C(C)C)NC(C(N1CC(O)(CC=C)C1)=O)CO 56676,c1(CN(C(=O)CC2(c3ccccc3)COC2)CC=C)cccc(F)c1F 56677,c1(CNC(=O)NC2CC(CSC)C2)ccc(N2CCOCC2)c(F)c1 56678,N1(C(c2c(C(C)C)cnn2C)=O)CCC(C)C(NC(=O)C=CCO)C1 56679,CN1CCC(Nc2cc(NCc3nc(C(F)(F)F)n[nH]3)ncn2)CC1=O 56680,c1(C(=O)O)ccc(C(N2CC(Cc3ccc(Cl)c(F)c3)C2)=O)c(F)c1 56681,c1(C(N2C3C(NC(c4c(CC)onc4)=O)CC(C3)C2)=O)c(C)ccc2n[nH]cc12 56682,C(CC(=O)NC(CO)C(N)=O)(C(C)(C)C)NC(C(C)n1cccn1)=O 56683,N1(C(C2OCCN(C(C)=O)C2)=O)CC2CCC1C1CN(C(c3ccsc3)=O)CC21 56684,C1(CNC(C2CC(NC(Cc3c(C)scc3)=O)C2(C)C)=O)CC2OC1C1CC21 56685,S(=O)(=O)(c1cc(F)c(F)cc1F)N1C(c2c(OC)cccc2)CC2(CCC2)C1.c1(C(=O)C=C)ccccc1 56686,N1(C(c2cc(C)c(F)cc2Cl)=O)CC(C)CN(C(c2ccc(N)cc2)=O)C(C)C1 56687,N1(CCN(C(=O)CC2(C)CC2(F)Cl)C)CCN(C(c2ccccc2O)=O)CC1 56688,c1(COC)nc(N2CC(O)(C(C)NC(C3CCN3C(C)(C)C)=O)C2)cc(O)n1 56689,c1(C(N(C2CCCN(C(CN(C)CC)=O)C2)CC)=O)cc2ccc(OC)cc2[nH]1 56690,C1(NC(COc2cccc(C)c2C)=O)CN(C(=O)Cc2cc[nH]n2)CCC1(F)F 56691,c1(CC(=O)N(C(C)CN(C(=O)C(O)c2ccco2)C)C)ccccc1C1CC1 56692,CC1CN(C(=O)CC(=O)Nc2nccs2)CC1CCNC(C1CC(C)(O)C1)=O 56693,C1(C(=O)NCCC(C)O)(OC)CCN(C(=O)C(O)C(C)C)C1 56694,N1(C(COC)=O)CCC(CNC(C2COCCN2CC(F)(F)F)=O)C1(C)C 56695,C(=O)(C1=CCCCCC1)N1C(CNC(C2CC(OCC)C2)=O)C(C)CC1 56696,N1(C(C(C=C=C)C)=O)CCC(C2CCN(C(c3ccc(=O)n(C)c3)=O)CC2)CC1 56697,C1(C(CC)CC)CC(C(N2CCN(C(=O)CCO)CC2)=O)CCO1 56698,c1(NC(C2CC(C)N2C(c2cc(=O)cc[nH]2)=O)=O)cn(C)nc1C1CC1 56699,C1(NC(c2ccc(CC)s2)=O)CC2CC(NC(C3(c4ccoc4)CC3)=O)C2C1 56700,C1(C(=O)NCC(CC)(C)C(N)=O)CC(C)(C)CCN1C(c1ccc(C(F)F)o1)=O 56701,C1(N(C(=O)CCC(=O)OC(C)(C)C)CC)CCCN(C(=O)C(C)CF)CC1 56702,N1(C(=O)COCc2nc[nH]n2)CCN(C(=O)Cc2ccc3c(c2)CC3)C2(CC2)C1 56703,CCC(CC(F)(F)F)C(=O)NC12CCCC1N(C(=O)C1=NNC(=O)C1)CC2 56704,Cc1ccc(C(N2CC3CC3(C(=O)Nc3nc(Cl)c(Br)nc3Br)C2)=O)c(I)c1C 56705,C=CC(C)CC(=O)NC1CCCC1CNC(c1cnc(C(F)F)cn1)=O 56706,CCCC(O)CC(=O)NC1(CF)CCN(C(=O)CN(CC)Cc2ccccc2)C1 56707,c1(NCCOC)ccc(S(=O)(=O)NC2CCC3CC23)cc1Cl 56708,c1cc(=NC2CCCSCC2)[nH]c(NCC2CCCOCC2)n1 56709,C(C)(C)(C(=O)N1CC(C(C(=O)NCC2(COC)CCC2)OC)C1)OC 56710,c1(OC)ccc(OCCC(N2CC(O)(CCNC(=O)C(C)=C(C)C)C2)=O)cc1 56711,N1(C(C2(C(=O)OC)CC2)=O)CCN(C(=O)COC(F)(F)F)C2(CC2)C1 56712,C1(=O)CC(C(F)(F)F)ONC(=O)C2CCCN12.C(=O)(C(F)(F)C(F)F)OC(C)(C)C 56713,c1(C(=O)OCC)nc(CNc2ncc(CC)s2)nc(-n2cccn2)n1 56714,CC1(CNC(=O)C(Cl)(Cl)Cl)CCN(Cc2cccnc2-c2cccc(F)c2)CC1 56715,C(C(C)C(F)C(=O)NCCC(F)(F)C(C)C)NC(c1cc(C)ns1)=O 56716,C1(N(C(CCC(=C)Cl)=O)C)CCCN(C(c2nocc2Br)=O)CC1 56717,CC(=O)C(C)(C)CC(=O)NCCOCCCNC(c1cc(C(N)=O)c[nH]1)=O 56718,C(=O)(C1=CCS(=O)(=O)C1)N1CCCC(CN(C(CC(CCC)C)=O)CC)C1 56719,c1(C(=O)NC2CC(NC(=O)CC3CCCC34CC4)C2)cc2ccc(Cl)c(F)c2o1 56720,C(=O)(C(CC(F)F)N(C)C(C1CCOC1C(C)C)=O)NCC(=C)CC 56721,C1(N2C(=O)C2C2CCCC2)CCSCC1.c1(CC2CCOC2)ccccc1 56722,C(=O)(C(C)(C)CC(C)C)N1CC(OCCNC(C(F)=CC)=O)C1 56723,Cc1ncc(C(=O)NC(C)C(C)(C)C(=O)NC2CN(C(N)=O)C2)c(=N)[nH]1 56724,C(=O)(CCC(F)(F)C(F)(F)F)N(CCC)CCNC(C1(C)CCOC1)=O 56725,C1(NC(C2N(C(CCC)=O)CCC2)=O)CC2CC1N(C(c1cc[n+]([O-])cc1)=O)C2 56726,c1(C(=O)NCC2C(C)CN(C(C3C=CCC3)=O)CC2)cc2cc(F)ccc2s1 56727,c1(C(=O)NCCCNC(CC)=O)ccc(CNC(=O)C(C)CN(C)C)cn1 56728,N1(C(C(C2CCCCC2)OC)=O)CCC2(NC(=O)C(C)O)CCCC12 56729,Cc1sc(Cl)c(C(=O)NC2CC2CNC(=O)C=CC(=O)N(C)C)c1C 56730,N1(C(C(CO)NC(C)=O)=O)CCC2CC(NC(C3CC3(C)Br)=O)CCC2C1 56731,c1(NC(C2CCCCC(c3ccccc3)C2)=O)ccc2c(c1)OCO2 56732,Cc1cc(C(C)(C)NCc2ncoc2C(F)F)ccc1F 56733,C1(C(N(CCCO)CC#C)=O)(OC)CCN(C(C2(C#N)CCCC2)=O)C1 56734,c1(C(=O)NCC(C)NC(c2c(NC)scn2)=O)cc(OC)cnc1F 56735,CC1CCCC(CCNC(C2CCN(C(=O)CCCc3cnn[nH]3)C2)=O)C1 56736,CCC(CC)CC(=O)NCc1ncoc1C1CN(C(=O)C(C)(C)C(C)C)C1 56737,Cc1cccc(C(=O)NCCOC2CN(C(C3(C(C)(C)O)CC3)=O)C2)c1F 56738,c1(C(=O)NCCC(C)NC(Cc2cncc(C)c2)=O)ccc2c(c1)CCC2=O 56739,C1(C(=O)NCCC(C)N(CCC)C)C=CCCN1C(=O)Cc1ccsc1 56740,C(c1ccc(Cl)cc1Cl)=CC(N1C(C(N2CC3CC3C2)=O)CC2CC21)=O 56741,N1(C(COCC(=C)C)=O)CCCC(N(C)C(c2ccc(Cl)s2)=O)CC1 56742,c1(NC(=O)CCc2ccc(-c3nn[nH]n3)cc2)ccc(F)cc1O 56743,c1(COC)cccc(C(=O)NC2CCCC(NC(=O)CSC(C)(C)C)C2)c1C 56744,C1(C)(NC(C(C)CC2CCC2)=O)CCN(C(=O)CCF)C1 56745,CC1(C)CC(C(N2CCCC(NC(=O)Cc3ccsc3)CC2)=O)CC(C)(C)S1 56746,C1(C(=O)OC)CC12CCC(NC(c1sc(SC)cc1C)=O)CC2 56747,c1(C(C(=O)NCCOCCNC(c2oc(C)c(CO)c2)=O)O)ccc(Cl)c(Cl)c1 56748,C12(CNC(=O)COC3CC3)CCC(CC1NC(=O)C(C1CCOCC1)O)C2 56749,c1(OC)cc(F)cc(F)c1S(=O)(=O)NC(C)(C)Cc1cc(F)cc(F)c1 56750,c1(-c2ccc(C(C)(C)O)cc2)cccc2c(C(=O)Nc3ncc(Br)s3)[nH]nc12 56751,N1(C(Cc2ccn(C)n2)=O)CCC12CCN(C(=O)COCc1cccnc1)CC2 56752,C1(C(N(CC(=O)OC)CCC)=O)CC12CCN(C(=O)CC(C)(F)F)CC2 56753,c1(C(c2n(CCC)nnn2)NCCCOC(=O)NC)c(Cl)cc(Br)cc1Cl 56754,c1(C(C)NC(CC(CC)(F)F)c2nnnn2CC2CC2)nnc2n1CCOC2 56755,c1(CC(=O)NCC2(F)CC(CNC(=O)C=CCN3CCC3)C2)csc2nccn12 56756,c1(C(=O)NCC2(COC)CN(C(C3CC4CC4C3)=O)C2)cnc2n1CCCC2 56757,C(CC(C(=O)NC(c1cn[nH]c1)C)NC(c1[nH]ccc1C)=O)OCC 56758,C(=O)(C(C)(F)C(=O)NCC(C)(F)CNC(=O)C(C)(C)c1cccnc1)OC 56759,S(=O)(=O)(c1ccc(I)cc1)N1CCN(C(c2ccc(NC)cc2)=O)CC1C 56760,N1(CN2C(C(CC)(C)C)CCC2)CCCC(C(=O)OC)C1=O 56761,C1(NC(C2CC23CCC3)=O)(CNC(C2CCCS2)=O)CC2CCC1CC2 56762,N1(C(C(CC=CC)C)=O)CC(NC(=O)C(C2(O)CCOCC2)(F)F)CC(C)C1 56763,C=C(C)CC(C)C(=O)NC1CCCCC1NC(=O)C(C)(C)CO 56764,Cc1ccc(CN2CC(CC(N3CCOC(C)C3)=O)C2)cc1[N+](=O)[O-] 56765,c1(C(=O)OCC(C2CC(=C)C2)=O)cccc(C2(C)CC2)n1 56766,C(=O)(C1c2c[nH]nc2CN1C(c1cc(CO)on1)=O)N(CCCC)CCCC 56767,S(=O)(=O)(c1ccccc1N)Nc1ccc(N(C)Cc2ccccc2)cc1 56768,CC(O)(CNC(c1coc(CNC(C2CC23CCCC3)=O)n1)=O)CCO 56769,c1(C(=O)Nc2ccc(NC(C3(CC)COC3)=O)c(C)c2)ccc2c(n1)CCC2 56770,C1(NC(c2cccc3ncsc23)=O)CN(C(c2cnco2)=O)CC12COC2 56771,c1(C(N(CC(C)NC(=O)CC2CCCCC23CC3)CC)=O)ccc(S(N)(=O)=O)s1 56772,N1(C(c2c(C(=O)OC)[nH]cn2)=O)CCC(C)(NC(c2cc(OC)cnn2)=O)CC1 56773,O=C(CCC(=O)c1cccnc1)NC1CCCC1NC(C1C2COCC12)=O 56774,c1(C(=O)NCCCCNC(C2C(C)CCOC2)=O)c(F)ccc(Cl)c1[N+](=O)[O-] 56775,C1(O)(C(C(=O)NC2CCC(C(=O)NC(C3CCCCC3)C)C2)N(C)C)CCCCC1 56776,C(C(=O)NC1CC(NC(=O)C(C)Sc2ccc(C)cc2)C1)(C(C)C)SC 56777,C1(NC(c2c(C)coc2C)=O)C2CCC1N(C(=O)Cc1cscc1Br)C2 56778,n1(CC)nnnc1C(c1nc(C(=O)OC)cs1)NC1CC1c1ccccc1 56779,C(C(=O)O)(C(C)C)OCC.CCC(C(=O)C(=O)NCc1nc(CN)sc1)C1CCC(=O)N1 56780,CS(=O)(=O)c1ccc(F)c(OC(=O)COc2cccc(C#N)c2)c1 56781,N1(C(c2scc(OC)c2)=O)CC(O)CC1(C)C(=O)NCc1ncccc1C 56782,N1(C(C2(CC)CCCCC2)=O)CC2(CC(NC(C3(O)CCC3)=O)c3nccn32)C1 56783,CC1(C)CC(C(=O)NCC(O)(CO)CO)CN(C(=O)Cn2cnnc2O)C1 56784,c1(-c2cccc(OCC)c2F)c(C(=O)NCc2cccn2C)[nH]c2ccccc12 56785,C1(=O)C(F)C(C)CNC2CC(C2)CC(=O)NC2CN1C2.N(C)(C)SC 56786,CC1CC(NC(C2COCCOC2)=O)CN(C(c2ccsc2)=O)C1 56787,N1(C(C2C=C(C)CS2)=O)CC2(C=C(C(=O)N3CCC(N(C)C)C(C)C3)CO2)C1 56788,Cn1ccc(C(=O)NC(C2CCOC2)CNC(c2n[nH]cc2Cl)=O)c1C1CCC1 56789,CCCC(C)CC(=O)N(CC(=O)N(C)Cc1cc(C)no1)C(C)C 56790,N1(C(CC(C)OC)=O)C2CCC(C2)C1CC(N1CC2(C=CCO2)C1)=O 56791,N1(C(=O)CC2CC3(C2)CN(C(c2cccc(F)c2O)=O)C3)CCCC2COCC12 56792,C1(N(C)C(C2CC(C(F)(F)F)C2)=O)CC(C)(NC(=O)CCNS(C)(=O)=O)C1 56793,C(=O)(C#CC1(C)CCCO1)NC(C1CCCN1C(c1cnccc1Cl)=O)(C)C 56794,c1(C(N2CC3C(CNC(c4cnc(C(C)C)s4)=O)C3C2)=O)ccc(Cl)c(F)c1N 56795,c1(N)cccc(Cl)c1O.CC(O)C=O.C1(C)C=CC(=O)N1CCO 56796,C(CCN=c1[nH]c(=N)[nH]c(=NC2CCCC(F)(F)C2)[nH]1)N1CCN(C)CC1 56797,Cc1snnc1C(=O)NCCC1CCC(NC(c2cnc(S)[nH]2)=O)C1 56798,N1(C(c2n(CC)ncc2)=O)CC2(C(=O)NC(COC)C(C)C)CCC1CC2 56799,C1(NC(C(C)(CO)NC(C(CN(C)C)N(C)C)=O)=O)CN(C)CC1(F)F 56800,C(C(C)(F)C(C)C)NC(c1c(CNC(CSCCC=C)=O)cco1)=O 56801,n1(CC(C)(C)CO)nc(-c2ccco2)nc1-c1cc(C2CC2)on1 56802,C1(CC(=O)NC(C)CC2CCC(O)(c3ccccc3)C2)CC(C)CC(C)(C)C1 56803,N1(C(c2sc(C)cc2C)C(=O)NCCC(=O)OCC)CCC(C#N)CC12CC2 56804,C1(C(N(C2CCN(C(=O)C=C3CCC(C)C3)CC2)CC#C)=O)COCC(C)(C)O1 56805,c1(CC)cc(CC(N2CC(F)(CNC(C3CC(F)(F)C3)=O)C2)=O)n(C)n1 56806,C1(CNC(CCCOCCOCC)=O)CN(C(C2CCNC2=O)=O)CC1C 56807,c1(C(=O)NCCN(C(=O)Cc2sccc2C)CCOC)nn[nH]c1Cl 56808,C=C(C)CCC(=O)N1CCC(NC(C2CC(C)=NO2)=O)C1CC 56809,C1(CNC(C2CCCC2F)=O)COCCN(C(C2CCCOCC2)=O)C1 56810,N(C(=NCc1ccc[n+]([O-])c1)NCc1nc(C(F)(F)F)cs1)C(C=C)C 56811,N1(C(c2c(C)n(C3CC3)nc2)=O)CCC(NC(=O)C2=COCCO2)CC1C1CC1 56812,C(=O)(C(CC(C)C)C(N)=O)NC(C(=O)N(CC#C)CCOC)C(C)C 56813,C(CNC(=O)Cn1ncc(Cl)c1C)(C(C)(C)C)NC(CCSCCCC)=O 56814,C(c1cccc(F)c1F)=CC(N1CCC(NC(c2cc(=N)[nH]cc2)=O)(CO)C1)=O 56815,N1(C(c2c(O)ncc(CC)c2)=O)CCCN(C(=O)CCOC)C(C)C1 56816,c1(CCC(N2CC(NC(C(CC)OC)=O)C(C(F)F)C2)=O)cnc2ccccn12 56817,Cc1cc(Br)c(C(=O)NC2CCC(F)(F)C2)cc1Br 56818,C1(NC(CC(CC)C2CC2)=O)CCSC12CN(C(=O)C(C)(C)OC(C)=O)C2 56819,CC1Oc2ccc(C(=O)NCC(=O)NC(c3ccccc3F)C)cc2NC1=O 56820,c1(C(=O)NCCCCCNC(C2(C)CC=CCO2)=O)nnn2c1CCC2 56821,c1(C(=O)NCC2C(NC(COCC)=O)COC2)cc2ccccc2cc1OC 56822,C1(C(=O)NC(C2CN(C(c3c(CC)c(C)sc3)=O)C2)C)CCC(N=[N+]=[N-])C1 56823,N1(C(C2C(C)C2)=O)CC(CNC(=O)Cc2nc[nH]n2)C2(CCC2)C1 56824,c1(-c2nc(-c3c(C(=O)OCC)cc(Cl)cn3)on2)cc(Br)c(O)cc1O 56825,C(=O)(C1CCc2nccn21)NCCC1(C)CCN(C(COCC(=O)OC)=O)CC1 56826,C(=O)(C1=NOC(CNC(=O)CCc2ccco2)C1)N1C(C#C)CCC1 56827,c1(C(=O)NC(C2CN(C(c3c(NC)cncc3)=O)C2)C)ccc2nc(O)cn2c1 56828,Nc1nonc1C(=O)NCC1(CC(N2CCC(F)C2)=O)CC1 56829,C1(CC#N)CCCN(c2ccnc(NCC3CC3c3cccnc3)n2)C1 56830,CCN(Cc1ccc(F)cc1)N1CCc2cc(CO)ccc2C1 56831,N1(C(C(c2ccccc2)NC(C(C)NC(C)=O)=O)=O)CC2C=CCC(C2)C1 56832,c1(C(=O)NC2COCCN(C(C3C4CCCCC34)=O)C2)c[nH]c2ccc(Cl)cc12 56833,Cc1cn(C)cc1C(=O)NCc1ccccc1CNC(=O)C(C)NC=O 56834,C(CCCCN(C)C(C12CCCC1C2)=O)NC(C1(C(=O)OCC)CC1)=O 56835,c1(C(N2C(C=CC(=O)N(CC(C)(O)C3CC3)C)CCC2)=O)cccc2ccnn12 56836,c1(C(N(C(=O)CS(C)(=O)=O)c2scc(C)c2)=O)cccc(C2CCOCC2)c1 56837,N1(C(c2c(C)nc(COCC)s2)=O)CCCN(C(C2(COC)COC2)=O)CC1C 56838,c1(C(C)(CO)N(C(c2cn(C3CC3)nn2)=O)CC2CC2)c(F)cccc1F 56839,c1(C(=O)NC2CC(NC(C#CC)=O)C2)ccc(I)c(C)c1 56840,C1(CC(=O)NCC2CCN(C(c3ncoc3C3CCC3)=O)C2)CC(=O)NC(=O)C1 56841,Cc1cc(C(=O)Nc2cnc(F)cc2C(=O)NC2CC(F)C2)nc2ccccc12 56842,N1(C(c2nc(C)sc2)=O)CCC(CO)(CNC(C2(N3CCCC3)CC2)=O)CC1 56843,CS(=O)(=O)c1ccc(F)c(C(=O)NCC2(F)CC(NC(=O)C(F)F)C2)c1F 56844,c1(C(N(C2CCN(C(=O)C(O)CN3CCCC3)C2)CC)=O)ccc(=O)oc1 56845,C#CC1CC2(CC(C(N3CCN(C(=O)C(C)(C)NC(C)=O)CC3CO)=O)C2)C1 56846,CC(C)CC(C)(CNC(C1(Cl)CC1(C)C)=O)NC(c1cccc(C2(C)CC2)c1)=O 56847,Cc1cc(C(=O)NCCOC2CCN(C(=O)Cn3cccc3)C2)cc2ccsc12 56848,CCC(C(=O)N1CCC(C(=O)N(CC(C)(C)O)C2CCC2)C1)C(C)(C)CC 56849,c1(OCC)cccc(C(N2CC(NC(C3CCC3(F)F)=O)CC2CO)=O)c1N 56850,C1(CNC(C2C(C)(C(C)C)C2)=O)CC2(CCC2)CN1C(c1c(F)ccnc1Cl)=O 56851,c1(C(N2CCCC(N(C(C(CC)N(C)C)=O)C)CC2)=O)cc2n(n1)CCNC2=O 56852,N1(C(c2nn(C)cc2Br)C(=O)NC(CC)C)CCCCC1C1OCCO1 56853,N(C=CC(=O)C(F)(F)F)C(=O)CC1CN(Cc2cc3ncccc3[nH]2)CCO1 56854,C(=O)(C(=O)CCC(C)C)NC(C(=O)N(CCCCC(=O)NC)C)CCF 56855,C1(NC(CN(CC(C)C)C(c2n(CC#C)cnn2)=O)=O)CCC2(CCC2)C1 56856,C#Cc1cccc(C(=O)NC2CC(CNC(c3cc(OC)n[nH]3)=O)C2(C)C)c1F 56857,c1(C2(COC(c3c(CS(=O)(=O)OC)onc3)=O)CCCC2)cccc(F)c1 56858,N1(C(C2CCC(C)C2)=O)CCOC2(CCN(C(c3cc(Cl)ccc3N)=O)C2)C1 56859,C1(CC(=O)NC2(C(N(CCOC)C)=O)CC2)CCC(C#N)C1 56860,c1(C(=O)NCC2(F)CC(CNC(COCCC(C)C)=O)C2)ccc(F)c(N)c1F 56861,CCCC(C(=O)N1CCC(NC(c2cncs2)=O)C(O)C1)C(C)C 56862,N1(C(c2c(C)ncs2)=O)CCC2(CCCC2NC(c2cc(O)nc(O)c2)=O)CC1 56863,N1(C(CC)=O)C2CCC1CN(C(c1c(C3CC3)cccc1C1CC1)=O)C2 56864,c1(CCC(=O)NC2CCC(NC(=O)CCC3CNC(=O)N3)C2)c(F)cccc1F 56865,c1(OCCC(=O)NC2(C)CCN(C(=O)CC3CC3)C2)ccc(F)cc1Cl 56866,c1(C(N2CCC(NC(C(C)OCC#C)=O)C(F)C2)=O)csc2cccnc12 56867,C1(CN(C)C)CCN(C(=O)C(O)CNC(c2ccccc2CC#N)=O)CC1 56868,CCC(CC)CC(C(=O)NCSc1ccccc1)N1CCCC(C)C1C 56869,C1(F)(CNC(c2ccn(C)n2)=O)CCN(c2nc(Cl)ncc2C2CC2)CC1 56870,C1(NC(C(C2CC=CCC2)NC(C)=O)=O)CC2(C1)CC(O)C2 56871,N1(CC(N2C(CN(C(c3cncnc3C)=O)CC)CCC2)=O)CCn2nccc21 56872,c1(CC(N2C(C(C(=O)NCCCC3CC(C)C3)(C)C)CCC2)=O)cccc(O)c1 56873,Cc1cc(=NCCc2ccc(C)c(F)c2)[nH]cc1S(=O)(=O)NC1CCS(=O)C1 56874,C1(CNC(C(C)OC)=O)CCC(NC(C2CCOC2)=O)CC1 56875,C1(NC(C2CC(F)CN2C(=O)Cn2ncnn2)=O)CCn2ncnc2C1 56876,C#CCC(CC(F)F)C(=O)NC(CNC(c1nccnc1C(N)=O)=O)CC(C)C 56877,Cc1cccc(C(C)OC(=O)C(C)OCC2CC2)n1 56878,N1(C(c2ccno2)=O)CCC2(CC1)CCN(c1ncc3ccccc3n1)CC2 56879,C(=O)(CC(C)(C)NC(C1COCCC1C)=O)NCC1(OCC)CC1 56880,c1(CC(=O)NC2CC(CC)(CC)N(C(=O)CNC=O)C2)cnn2ccccc12 56881,Cc1nn(C(C)C)cc1C(=O)NCC(CO)NC(=O)C(C(C)C)N(C)C 56882,Cc1ccnc(C(=O)NCCC(C)NC(=O)CC2CCC2(F)F)c1N 56883,S(=O)(=O)(c1ccc2[nH]c(=NC3CCN(CC4CC4)CC3)ccc2c1)NCCCC 56884,Cc1cncc(CC(N2CCC(n3cc(-c4cnc(C(=O)O)nc4)nn3)C2)=O)c1 56885,S(=O)(=O)(c1cccc2nsnc12)N1CC2(CCN(C(c3cnsn3)=O)C2)C1 56886,N1(C(C(N2CCNC2=O)C)=O)CCN(C(=O)COCC2(F)CC2)C(C)C1 56887,CCCC(C(=O)NC1CC2C(NC(c3[nH]nnc3C(F)F)=O)C2C1)OC 56888,C=C1COCCN(C(C2(N)CC=CCC2)=O)C1 56889,S(=O)(=O)(c1cc(C(F)(F)F)ccc1Cl)NC1CCN(C(c2cscn2)=O)CC1F 56890,N1(C(CC(C=C)C)=O)CCN(C)CC1CNC(c1ccn(CCF)n1)=O 56891,c1(OC)ccc(F)c(N)c1C(=O)NCC1C2CCC(C2)N1C(C1CC12CC2)=O 56892,N1(Cc2ccc(C(=O)OC)cc2)CCC(O)C(C(=O)Nc2cncc(Br)n2)C1 56893,C(=O)(C(CC(C)C)N(C(=O)C(C#N)C(C)C)C)NCCCn1c(C)ncc1 56894,C(CCN(C)C)(C(=O)NC1CCOC1CN(C)C)NC(C(c1ccncc1)C)=O 56895,CCCCCCC(F)C(=O)N1CCOC(C2CN(C(c3ccc(=O)n(C)n3)=O)C2)C1 56896,S(=O)(=O)(c1ccc(N(C)CCF)c(F)c1)N1CCC(OCC)CC1(C)C 56897,CCCCCC(O)CNC(=O)CC(CNC(c1c[nH]nc1C(C)C)=O)C1CCC1 56898,C1(NC(N(C2CN3CCC2CC3)C)=O)CN(C)C(C)(C)C1 56899,N1(C(CCNC(C(C)(C)C)=O)=O)CCC(O)C(NC(=O)Cc2csc(Cl)c2)C1 56900,N1(C(c2ccccc2F)=O)CCC2CCCC12C(=O)NCC1C=CCC1 56901,C1(CC)CN(C(C2CCOC2CNC(c2cccnn2)=O)=O)CCCO1 56902,c1(C(N2C(CC)CN(C(=O)C(CC)OC)CC2)=O)cc2ccccn2c1 56903,C1(C(=O)NCCN(CCCCCC)C(C)=O)(Cc2ccccc2)CCNC1=O 56904,C1(CC#C)(C(=O)N(CC(=O)N(CC(F)Cl)C)CC2CC2)CCOC1 56905,C1(c2c(C)n(C)nc2)C(C(=O)N(C)Cc2cnco2)CC(=O)N1C 56906,C(C)(C(CC(=O)NCC1CCCC1(C)C)NC(C1CCOC1)=O)OC 56907,c1(C2CN(CC(=O)N(C)C(=O)Oc3c(C(=O)OC)scc3)C2)cccc(Br)c1 56908,C1(C(=O)NC2CN(C(CCSCCCC)=O)C2)CCCN(c2cc(O)ncn2)C1 56909,c1(CCC(N2CC(O)(CNC(CCCOCC)=O)C2)=O)cccc(C(F)F)c1 56910,C(=O)(C(CC)C(C)C)NC(C(=O)N(CCOCC#C)C)CCC1CC1 56911,C(=O)(C1=NOC(C)C1C)NCC(CCOC)NC(c1ccc(C(F)F)c(Cl)c1)=O 56912,C1(CNC(CCCC(C)(C)C)=O)CN(C(=O)CCC2(C)N=N2)CCC12CCC2 56913,N1(C(c2ccc(OC)s2)=O)C2CCC1C1CC1(NC(c1cc(C)sn1)=O)C2 56914,N1(C(C(CCC)OCC)=O)CCC(CNC(c2cc(C(C)C)on2)=O)CC1C 56915,C(C(C)(CO)NC(c1sccc1NCCS(C)(=O)=O)=O)NC(C)=O 56916,C1(CNC(C2(OC)CCOC2)=O)CN(C(=O)CN(C)S(N)(=O)=O)C2(CCC2)C1 56917,c1(C(C(N2CCC(N(C(C(CC)F)=O)C)CC2)=O)(C)C)ccc(Cl)c(C)c1F 56918,N1(C(c2n(CC)ccn2)=O)CCC(NC(C2CCCN2C)=O)C(CC)C1 56919,C12(CNC(c3cc(COC)no3)=O)CCCC1N(C(C1CCC(=O)C1)=O)CCC2 56920,C(CC1=CCN(CC2CCS(=O)(=O)C2)CC1)NC(CCC(C)OC)=O 56921,c1(OC)cc(C(=O)NCCc2ncc[nH]2)ncc1-c1ccc(C)nc1C 56922,C(=O)(CCCCCF)NC1C(NC(C(N2CCCCC2=O)C)=O)CCCC1 56923,c1(N2CCCCC(NC(c3ccccc3)C)C2)cncc(S(C)(=O)=O)n1 56924,C(=O)(C1CCCc2c1ncn2C)NC1CC(C)(NC(CC=C(C)C)=O)C1 56925,c1(C(=O)NCC(CNC(C2CC2C(C)(F)F)=O)OC)cnc[nH]c1=N 56926,N1(C(c2n(C)nc([N+](=O)[O-])c2)=O)CCC2(CC1)CC(CNC(c1cocn1)=O)C2 56927,CCCCC(C(=O)NCCOOC(=O)C(=O)NCCCC)N(C)C 56928,N1(C(COCCOCC)=O)CCC2(CC1)CC(NC(C1CCCO1)=O)CO2 56929,c1(C(N(CC(CC)NC(=O)Cc2n[nH]c(C)n2)C)=O)cc(C2CCOCC2)on1 56930,N1(C(c2cc(CC)[nH]n2)=O)CCC(C)(C)C(C(=O)NC(C)Cc2cc(C)[nH]n2)C1 56931,C(=O)(C1=CC(O)CCC1)NC(C)C(C)(C)NC(C1SCCCS1)=O 56932,C1(C(=O)NCC2(C#N)CC2)CC2C=CC1N(C(C1CCCC(=O)C1)=O)C2 56933,C1(N(C(CCC(=O)N(C)C)=O)C)CCCN(C(c2ccc(O)cc2)=O)CC1 56934,c1(C(=O)NCC2C(NC(C(C)n3cnnn3)=O)C2)coc2cccc(O)c12 56935,Cc1c(CN2CC(C)CC2c2ccccc2F)cccc1F 56936,N(C1CCc2cc(Cl)ccc21)c1ccnc(NCC2CCN(CCOC)C2)n1 56937,N1(C(Cc2nc(=N)[nH][nH]2)=O)CCC(C(N2CC(C3CCCO3)C2)=O)(CO)C1 56938,CCCC(C)(CCC)C(=O)NC(C)C(C)C(=O)N1CCC(CC(N)=O)CC1 56939,N12CC(CC(F)(F)C1)C2=O.N1(C(c2cc(C(C)=O)[nH]n2)=O)CCCC(OC)CC1 56940,c1(NCC(C(C)C)O)ccc(S(=O)(=O)N2CCCC(O)C2)cc1F 56941,c1(OC)ccc(-n2nnc(C(=O)NC3CCC3NC(C3CC34CC4)=O)c2C)cc1 56942,CC1CC(C(=O)NC(C2CCN(C(=O)CC3CC3(Cl)Cl)CC2)C)=NO1 56943,Cc1c(CC(=O)NCC2(CNC(C3CC3C(N)=O)=O)CC2)cnn1C 56944,c1(C(=O)NCC2CC(NC(C(CCC)C#N)=O)C2)[nH]c2cc(Cl)ccc2c1C 56945,CCCCCCCN=c1[nH]c(=N)[nH]c(=NCc2cn(C(C)C)nn2)[nH]1 56946,C(=O)(C(C(C)CC1CC(F)(F)C1)N1CCC(OC(C)=O)C1)NC(CC)(C)C 56947,c1(C(=O)NC(C)C(=O)NCC2CC3(CCCO3)C2)cc(F)cnc1O 56948,S(=O)(=O)(C(F)(F)F)N1CC(NC(=O)CCc2cnc[nH]2)C1 56949,N1(C(CC(C)(C)O)=O)CC(NC(c2csc(Cl)c2)=O)CC(O)C1 56950,C(C1=CCN(C(c2ccc(N(C)C)nc2)=O)CC1)NC(C(C)SCC)=O 56951,N(C(=NCCC1COC(C)(C)C1)NCCF)CC(c1ccc(OC)cc1)(C)OC 56952,CC1CCCN(C(c2cncc(NS(C)(=O)=O)c2)=O)C1CCNC(=O)CO 56953,N1(C(C2(S(N)(=O)=O)CC2)=O)CC(NC(=O)Cn2cc([N+](=O)[O-])cn2)C(C2CC2)C1 56954,N#Cc1ccc([N+](=O)[O-])c(N(c2ncnc3[nH]c(Br)nc23)C(=O)C2CC2)c1 56955,C(=O)(CC(C)(F)F)NC(CN(C(=O)Cc1ccnc(C(F)(F)F)c1)CC)C 56956,C(=O)(C(F)(F)C=Cc1ccccc1)NCC(n1cc(C2(COC)CCC2)nn1)C 56957,C(=O)(CCC(=O)NN(C)C)N1CC(C)CC(NC(C2(c3cc(C)no3)CC2)=O)C1 56958,C(C(C)C)(C(O)C(=O)N1CC2(CC2)CC1C(=O)NC1CN2CCCC1C2)OC 56959,Fc1ccc(Cl)c(F)c1CNCc1cc(I)ccc1Br 56960,c1(OC)ccsc1C(=O)NCC(F)CNC(c1ccn(CC(F)(F)F)n1)=O 56961,C(=O)(CC(C)(C)C)NC1CC(C(C(=O)N(C)Cc2cnccn2)F)C1 56962,c1(OC)cccc2c1CN(C(C1C3CC(CC3F)N1Cc1ccc(C)s1)=O)C2 56963,C1(NC(c2c(C)cc(Br)o2)=O)COCCN(C(=O)C(C)O)C1 56964,c1(OC)ccc(C(=O)NCC(CNC(C2(C)SCCCS2)=O)CO)cc1N 56965,Cc1c(C(N2CCOCC2CCNC(=O)CC(C)N(C)C)=O)cccc1Cl 56966,c1(CCNC(=O)NCCP(C)(C)=O)nnc2c(=O)[nH]ccn12 56967,C1(C(=O)NCC)CCCN(S(=O)(=O)CC)C1.C1(=O)C(=O)NCCCN1CC 56968,N1(C(C(CC)N(CC)CC)=O)CC2=C(C1)CN(C(c1cc3n(c1)CCCC3)=O)C2 56969,C(=O)(C(CCCOC)NC(=O)CC(O)c1ccccc1)NCC1(CCC)CC1 56970,C1(CCc2occ(C(=O)NC(C(=O)NC(=O)C3CC3)C3CC3)c2)(CO)CC=CC1 56971,C1(NC(C2(NC(CC(C)O)=O)CC(O)C2)=O)CCN(C)C1=O 56972,Cc1c(C(=O)NCC(C)CNC(=O)COCC2CCOC2)ccc(F)c1F 56973,CC(C)C(F)(CNC(c1ccn(C)c1)=O)C(=O)NC1C(O)C2CCOC12 56974,C=CC1(C(=O)NCCC2CC(NC(C3C=C(C)CS3)=O)C2)CCOCC1 56975,c1(NC(=O)NC2CC(CCSC)C2)ccc2c(c1)OCCO2 56976,N1(C(C2C(C(=O)OC)C2)=O)CC(CNC(=O)CC(C)(C)SC)OC(C)(C)C1 56977,C1(CC)C(C(=O)NC2(CF)CN(C(c3cnc(C)nc3)=O)C2)CCN1C 56978,N1(C(C2N(C(CCC)=O)CCCC2)=O)CC2(NC(C3CCC3C)=O)CCC1CC2 56979,c1(C(=O)NCCCC(C)NC(C2C3COCC23)=O)cc2c[nH]cnc-2n1 56980,CCC(C)(C)C(=O)N1CCC(C(C)CNC(=O)Cc2csnc2C)CC1 56981,N#Cc1cc(Cl)cnc1N1CCCC(C(N2CCCC2C(=O)O)=O)C1 56982,C1(NC(C(n2c(C)ncc2)C)=O)CN(C(c2scnc2C(C)C)=O)CCC1F 56983,Cc1cc(CNC(c2coc(CNC(=O)C(O)C(C)(C)C)c2)=O)cnc1F 56984,N1(C(c2c(Cl)cc(C)s2)=O)CC(C)CCC1CNC(c1ccc(F)s1)=O 56985,CCC(C)CC(=O)NCC(O)CNC(C12CC(C(=O)OCCCSC)(C1)C2)=O 56986,C(CSC(C)(C)C)(C(=O)N1CC(CNC(c2csc(C)c2)=O)C1)NC(C)=O 56987,c1(CN2CCC(CC(=O)NCC3(C(=O)OC)CC3)C2)c(O)cc(F)cc1F 56988,C=CCC(C)C(=O)NC1CCN(C(c2ccc(-c3ccc(F)cc3)s2)=O)CC1 56989,C(=O)(C(C)(O)C(C)C)NC1C(NC(c2cc(C)sc2-n2cccc2)=O)CCCC1 56990,c1(NC(C2CC(NCc3ccc(C)cc3Br)C2)=O)ccc(C#N)c(Cl)c1 56991,N1(C(c2nc(C(C)C)sc2)=O)CC(NC(=O)C2=CCSC2)C2(CCC2)C1 56992,C1(NC(c2cc(CNC(CC(C)C)=O)[nH]n2)=O)CCCC1(C)C 56993,N1(C(C2(C(F)(F)F)CCNC2)=O)CCC(F)(C(=O)O)C1 56994,C(CC)(CC)(CCNC(c1cccc(Cl)c1F)=O)NC(C(CC)n1ccnc1)=O 56995,N1(C(CC(=O)NCC#C)=O)CCC(C)(C)C1C(N1CCC1(C)CCO)=O 56996,c1(NC(C(C(C)C)NC(CCC=C)=O)=O)cnc(Cl)nc1C 56997,C1(OC)CN(C(=O)CC2CCOCC2)C(C)(CO)C1.c1(C=O)cc(C(N)=O)[nH]n1 56998,C(C(C1CCCCC1)NC(=O)CCF)(C(C)C)NC(c1ccc(SC)s1)=O 56999,C=CCC(C)(CC)C(=O)NC1CN(C(C2(O)CCOCC2)=O)CC2(CC2)C1 57000,N#Cc1ccc(CCNCc2nnco2)cc1 57001,c1(NCC(c2ncc[nH]2)C)[nH]c(=NCC2CC(C(F)(F)F)C2)nc2c1ncn2C 57002,n1(CO)cc(C(=O)NC2CCC(NC(C(C3CC3)SC)=O)CC2)c(O)nc1=O 57003,c12cn(nn1)CCCS2.c1(C(N(CC(=O)NC(C)C)C(C)C)=O)cnn(CCF)c1 57004,c1(CC)[nH]ccc1C(=O)NC(CC1CC1)C(=O)NCC1CC1(F)F 57005,c1(NC(N2C(C=NC(c3cc(OC)no3)=O)CC2)=O)ncnc2sccc12 57006,c1(C(=O)NC2C(OC)CN(C(=O)C(CO)N(C)C)C2)cc2cc(Cl)ccc2n1C 57007,n1(CC)cc(C(F)(F)C(=O)N2CC(C(C)NC(=O)C(C)(C)c3cscn3)C2)cn1 57008,c1(COC)ccc(NC(C2CN(C(=O)CCc3ccc(F)nc3)CCS2)=O)cc1 57009,c1(C(C)C)cnc(N2CC(C(=O)Nc3ncncc3Cl)C2)c(Cl)c1 57010,N1(C(CCCOCC)=O)CCCC(CN(C(=O)C(n2cc(Cl)cn2)C)C)C1 57011,N1(C(C(C)O)=O)CCCC(C2CN(C(C3CCc4n[nH]cc4C3)=O)C2)C1 57012,c1(N2CCC(NC(C3CCCSC3)=O)C(F)C2)nc(Cl)nc2[nH]ccc12 57013,C1(CCC)C(=O)NCCN1C(=O)NC(c1ccncn1)C 57014,C1(CCOC)(NC(=O)CC(C)(C)C2CC2)CCN(C(c2coc(C(F)F)c2)=O)C1 57015,N(C(=NCc1coc(C)n1)N1CCC(Cc2ccccc2)C1)C(C=C)C 57016,Cc1cc(N2CCN(C(=O)C=CC(C)(C)C)C(C)C2)nc(-c2cccnc2)n1 57017,C12(NC(=O)C=CC(F)(F)F)CC(CNC(=O)C=CCOCc3cccnc3)(C1)C2 57018,C1(C(c2nnnn2C2CC2)NCc2ccsc2)CC2(CCC2O)C1 57019,N1(C(N)=O)CCC(NC(=O)Nc2cccc(CSCCCl)c2)CC1 57020,c1(C(=O)NC(CN(C(COCCC=C)=O)C)(C)C)cc2ccccc2nc1O 57021,Cc1cc(C(=O)NCC2CC(F)(CNC(C3(C)CC3(F)Cl)=O)C2)ccn1 57022,c1(OC)ccc(C(=O)C(N2CC3CC3C2C(=O)NOCC(O)CO)=O)cc1Cl 57023,c1(C(C)C)ccc(C(N2CC3C(NCc4ccc(I)cc4Br)C3C2)=O)c(Cl)n1 57024,CC1COCCN1CCNC(C1CC12CC(NC(=O)Cc1ccc(O)cc1)C2)=O 57025,CP(C)(=O)C(O)C(=O)N1CCC(CCCCNC(C2CCC(=O)O2)=O)CC1 57026,NS(=O)(=O)CCCC(=O)N1CCN(C(=O)CCCN2CCCCC2)C2CC12 57027,c12cc(ccc1OC)CO2.c1(C(=O)Nc2n(CC#C)ncc2)ccc(C)cc1Cl 57028,c1(OC)c(F)cc(C(=O)NC2CCC2NC(=O)CC2CC(C)(C)CO2)c(N)c1F 57029,N1(C(C2(C3CC3)CN(C(C(C3CC3)SC)=O)C2)=O)CC(C2=NOCC2)C1 57030,CC12CCCC1N(C(=O)C1=NOCC1)CCN(C(=O)CCC1CCCCCC1)C2 57031,c1(OC)c(C(=O)NC23COC(C2)C(OC(C)C)C3)nc(O)nc1O 57032,C1(=CC(=O)NC2CCC(CNC(Cc3ccn(CC)n3)=O)C2)CN2CCC1CC2 57033,C1(C(N(C)CCC2CCCCN2C(=O)C(Cl)=CCl)=O)OC2CCC1CC2 57034,C(=O)(C(F)(F)C(F)F)N1CCC(CNC(c2ccsc2)=O)CC1 57035,c1(C(=O)NC(CC)CNC(=O)C(C)N(CC)CC)cc(F)ccc1C(F)(F)F 57036,C#CCC(CCCO)NC(C1CCCC1NC(C1CC2(C1)CC21CC1)=O)=O 57037,c1(C(=O)NC2CC(NC(CCC#C)=O)C2)ncn2c1COc1ccccc1-2 57038,c1(SCC(=O)NC2CCN(C(C3CCCC3O)=O)C2)n[nH]c(O)n1 57039,C(=O)(CCC(=O)NC1C2CC1N(C(=O)C(C1CCCCCC1)C)C2)NCCC 57040,C1(C(=O)NCC(CNC(=O)CC2(NC(C)=O)CCC2)OC)CC(C)CC(C)(C)C1 57041,c1(NC(N2CCC(CC3CCC3)C2)=O)ccc(C(F)(F)F)cc1O 57042,CCCC(CC(C)C)C(=O)NC1CCC(CCNC(=O)C(C)(C)n2cnnn2)C1 57043,c1(NC(C2(NC(C=CCOC)=O)CC(F)C2)=O)ccc(F)cc1C 57044,C(CC(C)(C)CC(=O)N1CC(NC(c2cn(CCO)nn2)=O)CC1C)OC 57045,C=CCC(CN(C(C)CC)C)C(=O)N(C(=O)CCC(=O)N(C)C)C 57046,c1(C(=O)NCC(CC)NC(=O)C(c2cccnc2)C)nn(C)c(Cl)c1Br 57047,N1(C(C2CCN(C)S2(=O)=O)=O)C2CCC1CN(C(C1CC(CCO)C1)=O)C2 57048,Cn1cc(Cl)c(C(N2CCC(Oc3cnccc3CNC(=O)C(C)(C)F)C2)=O)n1 57049,N1(C(Cc2c(C)n[nH]c2)=O)CC2CCN(C(c3cccc4nscc34)=O)CC2C1 57050,CC(C)C1=NOC(C(=O)NCCOCCNC(=O)Cn2cc(Br)cn2)C1 57051,Cc1cc(NC(=O)NC(Cn2cc(C(C)(C)O)nn2)CC(C)C)c(C)s1 57052,CC1CCC=C1C(=O)N1CCOC(CCNC(=O)Cn2ccc([N+](=O)[O-])n2)C1 57053,c1(CNC(C2C(C(C)C)CCO2)=O)cnn(C)c1C(=O)NC(C(C)C)C1CC1 57054,C1(C(N2CC(F)(C(=O)NC3(C(N(OC)C)=O)CC3)C2)=O)CC12CCOC2 57055,N1(C(c2ncnc(C)c2C)=O)CC2CCCC1C2CNC(c1ccc(F)cn1)=O 57056,c1(-c2nc(COC)nn2-c2c(CO)cc(Br)cc2C)noc2c1CC(C)CC2 57057,CC1(C)CCC(C(N2CCCC(CNc3ccccn3)C2)=O)C1 57058,C(=O)(CCCCCCCBr)NC1C(C(=O)Nc2c(C(=O)OC)cccn2)CCC1 57059,C(C)(C)(C(C)CC(=O)N1CC(C)CC(O)C1)NC(C(C)OCCN(C)C)=O 57060,C1(CNC(=NCCC)NCCC2CCOCC2)CCC2(CCCC2)O1 57061,CC(O)CCCNC(=O)CC1CCCC1NC(=O)Cc1ccsn1 57062,c1(C(N2C(C(C)NC(Cc3c(C)con3)=O)CCC2)=O)cn(C)c(=O)cc1Cl 57063,N1(C(C(CC)SC)=O)CCCC2(CCN(C(C)C(=O)N(C)C)C2)C1 57064,c1(CNC(C(N)=O)CO)cccc(OCC(F)F)n1 57065,c1(C(=O)NC(CNC(CSCC(=O)OC)=O)CO)ccc2c(c1)CCCS2 57066,C(=O)(C(O)CC(C)C)N1CCCC(CN(C(C2CN(c3nncs3)C2)=O)CC)C1 57067,c1(C(N2CCN(Cc3cnc(CCCC)[nH]3)C3C2C3)=O)ccc(F)c(OC)c1F 57068,C1(c2cn(Cc3c(CC)ccs3)nn2)C(C)CCN1C(=O)C(C)N1CCC1 57069,c1(C(=O)NCC(C2CCOC2)NC(C2(CC)CC2)=O)ccnc2ccc(F)nc12 57070,N(C1CN(C(c2cc(C)c(Cl)c([N+](=O)[O-])c2)=O)Cc2ccccc21)C(C)=O 57071,c1(C(=O)NC2C3CN(C(c4c(C)nn(CCO)c4)=O)C2C3)ccc2occc2c1 57072,C1(CC(=O)NC(C2(C(=O)NCC(C)Cn3ccnc3)CC2)C)CCCCO1 57073,Cc1cc(-c2cc(C)ccc2F)ccc1CN(CC(C)(C)CO)C 57074,C1(NC(c2c(OC(C)C)n[nH]c2)=O)CCN(C(c2n[nH]cc2Cl)=O)C12CC2 57075,C(=O)(C(C)C(C)C(C)(C)C)N1CC(OC)(CNC(=O)CCF)C1 57076,C(=O)(C(O)C(C)(C)CC)N(CCNC(C1N(CCC)CCC1)=O)C 57077,C1(CC=C)N(c2ncnc(NCCC(O)C(C)C)c2C)CCCC1(C)C 57078,Cn1ncc2nc(Cl)nc(N3CCC(NC(=O)CCC(N)=O)C34CCC4)c12 57079,C1(NC(c2sccc2Cl)=O)CCN(C(C2CC(C3CC3)C2)=O)CC(O)C1 57080,C(=O)(C(C)C(C)(C)C)N1CCC(C2N(C(C(C)SC)=O)CCCC2)C1 57081,c1(C(=O)NCC2CC(NC(C3C(C)C3)=O)C(O)C2)cc([N+](=O)[O-])c(F)cc1N 57082,CC1CCN(C(c2cnc(N)c(CO)c2)=O)CCN1C(=O)CCc1cnn(C)c1 57083,c1(C(N(CCC(C)NC(C2(CO)CCOC2)=O)C)=O)cc(Cl)ccc1N 57084,C(=O)(C#CC1CCCCC1)N1C2CN(C(c3c(NC)nccc3)=O)C(C2)C1 57085,C1(NC(=O)CCN(C(C2CCCCC2O)=O)C2CC2)CCC2CCCC1O2 57086,N1(C(C2CCC(NC(C3CCC(C)(CC)O3)=O)C2)=O)CC2CCCCC12C 57087,c1(-c2c(C(=O)NC(C(C)NC(CCCC)=O)C)c[nH]n2)ccc(Cl)cc1 57088,N1(C(C2(CC)CCC2)=O)CCC2(CCOC2)C(CNC(=O)CCC2(O)CCC2)C1 57089,C(=O)(CCCCCSC)NCC1(C(=O)NCC(C(CC)C)C)CCC1 57090,CCC(CC(=O)N1CCCC1CCNC(=O)C=C1CCC1)SC 57091,C#CCC(O)C(=O)N(CC(=O)NCc1ncsc1C)CCC 57092,C1(C(C)(C)NC(C=CCOC)=O)CCCN1C(=O)C(n1nccc1C)C 57093,N1(C(CCN(C)CC)=O)CCC(NC(C2(C)CC(O)CN2C)=O)C(F)C1 57094,C1(C(=O)NCC2(SCC)CC2)CNC(=O)CN1C(=O)C=CC1CCCN1C 57095,C(=O)(CS(=O)(=O)CC(=O)N1CCN(C(=O)C(C)N(C)C)CC1CF)OC 57096,C(=O)(C#CC(C)(C)C)NCCOC1CCN(C(c2nn(C)c(Br)c2)=O)C1 57097,C1(CNC(=O)COC2CCC2)CC2(CO1)CN(C(C1CCC(=O)O1)=O)C2 57098,c1(CN(CC(=O)N(C)CC2CCN(C(CCSC)=O)C2)C)ccc(Cl)cc1 57099,CN=c1[nH]cc(C(N2CC(O)CC2C(=O)NCC2COC(=O)N2)=O)o1 57100,C1(NC(C2CCC(CCC)CC2)=O)CN(C(=O)C(C)(C)O)CCC1(F)F 57101,C1(C(=O)NC2CN(C(c3ccn(C)c3)=O)CC23CC3)CCC2(CC1)CNC(=O)C2 57102,C(=O)(CC(C)C(=O)N1CCC(CNC(c2cnc(S)n2C2CC2)=O)CC1C)OC 57103,C1(C(N(C(C(=O)NC(N)=O)C2CC2)C)=O)OCCCC1(C)C.C12(CC1)C(=O)N2 57104,N1(C(C2N(CC)CCC2)=O)CCCCC1CNC(=O)Cc1cccnc1Br 57105,Cc1ccc(S(=O)(=O)N2CC(NC(c3c(C(F)(F)F)cccc3F)=O)C2)cc1C 57106,CCC(O)C(C)(C)C(=O)NCCCN(C)C(c1csc(-c2ccc(Cl)cc2)c1)=O 57107,C(=O)(C(C)(CO)NC(C1CC(C#N)(OC)C1)=O)NCc1n(CC)ncn1 57108,Cc1nc(C2CCCO2)sc1C(=O)NC1COCC1NC(c1ccccc1O)=O 57109,N1(C(=O)OC)CCCC(C(=O)NCC=CCNC(=O)CC2CCCC23CC3)C1 57110,c1(C(N)=O)cc(Cl)ccc1NC(=O)CCC1CNC(=O)N1 57111,C1(NC(C2CCN(C(C#C)=O)C2)C(=O)N(C)C)CCC(C(=O)NC)CC1 57112,C1(O)(CNC(C(C)C2CC2)=O)CC2CCC(C1)N2C(c1cnc(S)nc1)=O 57113,N1(c2ccnc(NCc3ccc(F)c(C)c3F)n2)CCCC2(CC1)CNC(=O)C2 57114,N#Cc1cc(S(=O)(=O)N2Cc3c[nH]c(=N)nc3C2)ccc1NCC1(F)CCOC1 57115,C1(C)(NC(C(C)C2CCCO2)=O)CCN(C(c2cc(N)cc(O)n2)=O)CC1 57116,C1(C(=O)Nc2ccc(-n3cccc3)nc2)CN(C(C2CC23CC3)=O)CC12CC2 57117,CC1OCCN(C(C2CC(=O)CN2C(=O)CCc2ccoc2)=O)C1C 57118,N1(C(C(C)OC2CCOC2)=O)CC2CC1CN2C(C1CC(C)(C)CN1C)=O 57119,C1(CC(=O)NCC(CC=C)NC(c2sccc2C)=O)CCCC(C)(C)CC1 57120,C1(NC(C(C)C2CC2)=O)CCC2(CC1)CN(C(=O)Cc1csc(S)n1)CCO2 57121,Cc1cccc(C)c1CC(N1CCC(CO)C(NC(c2[nH]cnc2C#N)=O)C1)=O 57122,N1(C(C(C(CC)C)O)=O)CCN(C(=O)CCCNC(=O)C(C)(C)C)C2(CCC2)C1 57123,N1(C(C(C)OCC)=O)CCC(N(CC(C)C)C(c2cccnc2C2CC2)=O)CC1 57124,N1(C(C(C)C#N)=O)CCOCC1CC(=O)N(C)CC1(O)CN(C)C1 57125,C1(NC(CCCC)=O)CCCN(C(=O)C=CCOCC(F)(F)F)C1 57126,C1(C)(CCCC(C2CCN(Cc3c(C)cncn3)CC2)=O)NC(=O)NC1=O 57127,C12(CNC(C(C)(C)F)=O)CN(C(c3ccc(OC(F)F)cc3F)=O)CC1CCO2 57128,c1cc2c(CNCCC3CCOCC3)[nH]c(=NCCC(O)C3CCCC3)sc-2n1 57129,n1(CC(=O)NC2CCCN(C(C3N(CC)CCC3)=O)C2C)ncc2cccnc12 57130,C(c1ccc(C(F)(F)F)cc1)=CC(N1CCNCC1C1CCCC1)=O 57131,N1(NCCCNC(=O)CC2CC23CC3)CCN(c2cc(Cl)ncn2)CC1 57132,N1(C(CC2(C)CC2)=O)CCC2(CCCC2NC(c2[nH]nc([N+](=O)[O-])c2Cl)=O)C1 57133,CCCC(CN=C(NCC1(CO)CC2CCC2C1)NC1CCC1)OC 57134,c1(C(=O)NC2(CC)CC(F)(F)C2)ncc(NC(=O)COC(C)C)cn1 57135,CC(C)C(CNC(=O)CCC1CCCCO1)NC(=O)CCCN(C)C 57136,C1(C(CC)O)CCCN1C(=O)C=CCNC(=O)CC1(COC)CC1 57137,c1(OC)cccnc1-c1cn(C2(C(=O)NC(C)CC3CCOC3)CCC2)nn1 57138,N1(C(CSS(C)(=O)=O)=O)CCCN(C(=O)C2CC2)CCC1.C12CC(C1)C(=O)NC2=O 57139,O=C1CCOC(C(N2CCCC2c2cn(CC3COCCO3)nn2)=O)C1 57140,C1(NC(=O)OC)CCCN(CCC(=O)CCOc2ccc(C(C)(C)C)cc2)C1 57141,C1(CCC)CN(C(=O)C(C#N)CC)CCN1C(c1ccnc(O)c1)=O 57142,N1(C(C2(CCC=C)CN(C(=O)C(O)C(C)C)C2)=O)CC(C)(C)C1COC 57143,N1(C(C=C(C)C)=O)CCN2CCN(C(=O)CCc3ccccn3)CC2C1 57144,CC1(CNC(=O)CCC2CNC(=O)N2)CCCN1C(c1cc[nH]n1)=O 57145,c1(C(=O)NCC2N(C(C(COC)C)=O)CC2)nc(-c2ccco2)oc1C(C)C 57146,CC(C)C#CC(=O)NCCCCNC(=O)CC(C)NC(C1CCCC1)=O 57147,c1(CCC(=O)NC(C2CC=CCC2)C(=O)NCCC(C)N2CCCC2)nncn1C 57148,C1(C(N2CC(NC(c3cc(C)[nH]n3)=O)C3C(C2)C3)=O)CN2CCCN1CC2 57149,c1(N2CCCC(CCNC(CSC(C)C)=O)C2)ccc(C#N)cc1[N+](=O)[O-] 57150,Cc1ncc(Br)c(N2CCC(C(N3CC(O)C(O)C3)=O)C2)n1 57151,C(=O)(CCCCC(=O)Oc1cccc(CC)c1)N1C2C(=CC)C(C2)C1.C1C(=O)N1 57152,Cc1nscc1C(N1CC=CC1CNC(c1cc(C(C)(C)C)n[nH]1)=O)=O 57153,C1(OC)CN2CC1NC(=O)C1(CCCC1)C2=O.C1(C)(CN(C)C)CCOCC1 57154,c1(C(COC(CNC(C2C(C)CCC2)=O)=O)N(C)C)cccc(C(F)(F)F)c1 57155,C1(C(=O)NC2C(C(=O)OC)CCC2)CCCCN1C(=O)Cc1ccoc1 57156,C(=O)(CC(C)CC(=O)N1CC(=O)CC1C(N1CCOC(C2CC2)C1)=O)OC 57157,C1(C(N(CC(N)=O)CC)=O)CCC(C)(C)N(C(C2CC=CCC2C)=O)C1 57158,c1(C(N2C(C)(C(=O)Nc3cc(C)cc(F)c3)CC2)=O)cnc2ccccc2c1 57159,C1(CC)(NC(=O)CCC2CCCO2)CCCN(C(c2ncc(OC)cc2F)=O)C1 57160,CC1=C(C(=O)N2CCC(F)(CNC(=O)CC3CCCCC3(C)C)C2)CCO1 57161,Cc1nnc(O)c(C(=O)NCC(O)CN(C(=O)Cc2cn3ccsc3n2)C)c1C 57162,CC1(C)CC(CNC(=O)CNC(=O)C(C)(C)C)N(C(C2SCCCS2)=O)C1 57163,c1(CC(=O)NC(CC(C)C)C(=O)OC(C)(C)C)c[nH]c2ccccc12 57164,CC1CCN(C(c2cccc(SC(F)F)c2)=O)CCN1C(C1CCCC(=O)N1)=O 57165,c1(CCC(=O)N(CCNC(=O)Cc2cc[nH]c2)CC)c(F)cccc1F 57166,C(=O)(CC(C)(C)C#N)NCC1C(C(=O)NC2CCN(CC)CC2)C1 57167,N1(C(C2CC(C#C)(O)C2)=O)CCC(C)C(NC(C2CC(C(C)C)C2)=O)C1 57168,CC(c1ccccc1F)=CC(=O)NC1CC(NC(C2(F)CCCC2)=O)C12CCC2 57169,N1(C(C(C)(C)c2ccccn2)=O)CCC2C(C1)CN2C(c1c[nH]c(C(N)=O)c1)=O 57170,c1(C(N2C(CNC(C(C)SCCCC)=O)CC2)=O)ccccc1[N+](=O)[O-] 57171,CC(C)C(C(C)NC(=O)Cn1cnccc1=O)NC(=O)CCn1cnccc1=O 57172,CN1CCN(C(C2(C#N)CCSCC2)=O)CC1CNC(=O)Cc1cncs1 57173,CC1(C)CCC(O)(CNC(c2ccc(CNC(=O)CC3CC3(C)C)nc2)=O)C1 57174,C(=O)(C(C)(C)C(=O)NCC(C)(O)CCO)NC1C(C(=O)OCC)CC1 57175,c1(N2CC(C(N3C(C)CCCC3C)=O)C(O)CC2)ncc2[nH]ccc2n1 57176,N1(C(CNC(CC(C)C)=O)=O)CC2C(CNC(C3CC4C=CC3C4)=O)C2C1 57177,c1(C(N2CCC(O)(C(C)NC(CC=C=C)=O)C2)=O)[nH]c2cc(OC)ccc2c1C 57178,c1(C(=O)NC(C2CCCN2C(=O)CN(C2CCSC2)C)C)nnnn1C(C)(C)C 57179,Cc1[nH]c2ccccc2c1C(=O)NC(C)CN(C(=O)CC1CC(F)C1)C 57180,C1(C)(C(=O)NCC(CNC(c2ccc(C(C)C)nc2)=O)O)CC(C(F)(F)F)=NO1 57181,C(=O)(C1CCCn2cncc21)Nc1c(OC)cccc1 57182,Cc1ccc(C(=O)NC2CCN(C(=O)Cc3nc(=N)[nH][nH]3)C(C)C2)cc1C1CC1 57183,N1(C(CS(=O)(=O)NC)=O)CC2(CCN(C(C34CCN(CC3)CC4)=O)CC2)CC1C 57184,Cc1cc2[nH]c(C(N3CCCC(NC(c4cc(F)n(C)n4)=O)C3C)=O)cc2o1 57185,c1(C(=O)NC(CCN(C(C(C)O)=O)C)C(C)(C)C)c(C(F)F)nc2cnccn12 57186,C(CCCCNC(c1cnn(CC(F)(F)F)c1)=O)NC(=O)Cc1cncnc1 57187,C1(NC(C(C2(O)CCCCC2)CC)=O)CCN(c2cc(C(F)F)ncn2)CC1O 57188,c1(C(=O)NC2CCC(NC(Cc3cc(C)ns3)=O)C2)ccc(-n2cncn2)cc1 57189,CCCC(CC)CC(=O)NCC1(NC(C23CCC(N=[N+]=[N-])C2C3)=O)CCCCC1 57190,c1(CNC(C(CCC)O)=O)cccc2c1CN(C(c1sc(CO)nc1C)=O)C2 57191,c1(CCCC(=O)NCCN(C(C2C(C=C)C2)=O)C)ccccc1Br 57192,Cc1nn(C)c(Br)c1C(N1CCCC(N(C(=O)CCOC2CC2)C)C1)=O 57193,C(=O)(CCCC(C)(C)CC)N1CC2C(CNC(c3ccc(C=C)cc3)=O)C2C1 57194,C1(NC(C2C(C)(C)C2)=O)C2CC1CN(C(C1CCN(c3nccs3)CC1)=O)C2 57195,c1(C(=O)NCC2OCCN(C(c3[nH]cc(C(C)(C)C)c3)=O)C2)nccc(Cl)c1Cl 57196,c1(CC)cc(C(=O)NC(CN(C(=O)CN2CCCC2=O)C)CC)ccc1C 57197,C1(NC(=O)COC2CC(F)(F)C2)CCN(C(c2csc(O)n2)=O)CCC1CO 57198,N1(C(CN(CCC)C)=O)CCC(O)(C(C)NC(c2cc(Br)cn2C)=O)C1 57199,O=C(C1=NOC2(CCC2)C1)NC1CC1CNC(=O)COc1c(Cl)cccc1Cl 57200,C1(NC(C2(OCC)CCSCC2)=O)CN(C(=O)CSc2cnn(C)c2)CCC1F 57201,C1(C)(C(N(CC(C)OC)C)=O)CCCN1C(c1ccc(CO)s1)=O 57202,n1(CC)ncc(C(N2CCOCC2CC(N2CC(O)C2)=O)=O)c1C 57203,CC(C)CCCC(C)NC(C1CC2(C1)CN(C(c1cccc(F)c1O)=O)C2)=O 57204,C1(CNC(C(C)OCCC(C)C)=O)(CNC(=O)C(N)=O)CC1(F)F 57205,CCCCCCCC(=O)N1C2CCC(C2)C1CNC(C1CCCS(=O)(=O)C1)=O 57206,CCCCCCCCC(C(=O)NC1COC1)N1CC2CSCC2C1 57207,C=C(C)CC(C(=O)N1CCC2(CC2C(=O)NCCCc2ccccn2)C1)OC 57208,C(CS(=O)(=O)CC(=O)NC1C2CC1N(C(C1CCc3nc[nH]c3C1)=O)C2C)OC 57209,c1(C(CNC(CCNC(C)=O)=O)NC(=O)C(O)C2CCC2)ccccc1F 57210,c1(C(=O)NCC2CC(NC(c3c(CC)cno3)=O)C2)ccc(Br)c(N)c1 57211,C1(CC(=O)NCC(CNC(c2c(C(=O)OC)csc2)=O)CO)CC=CCN1C 57212,CCC(C(=O)N1CCC(CC)(NC(=O)CCc2ccccc2Cl)CC1)C(C)C 57213,c1(OC)ccnc(F)c1C(N1CC(CNC(=O)C(C)SC(F)(F)F)(OC)C1)=O 57214,N1(C(c2c(COC)ccs2)=O)CCN(C(=O)C(F)C(C)(C)O)CC12CCC2 57215,CCC(CCCO)NCc1cccc(OCC(F)(F)F)c1 57216,CCC(CC)(CO)C(=O)NCC1CCC2(CN(C(c3ccnc(C)c3O)=O)C2)O1 57217,N1(C(C(P(C)(C)=O)O)=O)CC2(CCN(C(=O)CCn3cccn3)C2)C1 57218,Cc1cc(C(=O)NCC(=O)NCC2(C(N)=O)CN(C(=O)C(C)(C)CF)C2)c(C)o1 57219,c1(CC(=O)NC2CC(C(N3CC(C)OCCC3)=O)C2)cnc2ccccn12 57220,c1(C(=O)NC(C(C)(C)NC(C(C)NC(C)=O)=O)C)c[nH]c2ccc(F)cc2c1=O 57221,C1(NC(C2C(OCC)C2C)=O)CCCN(C(=O)C(C)=C(C)C)C1 57222,C(=O)(CC1=NNC(=O)C1)NC1CN(C(c2cc(C)nc(Cl)c2)=O)CC1C 57223,C1(NC(CN(S(CC)(=O)=O)C)=O)CCN(C(C2CC2C2(C)COC2)=O)C(C)C1 57224,C(C(C(C)C)OC)(c1n(CCSC)nnn1)NC1C(Oc2ccccc2)CC1O 57225,C(=O)(C(C)S(C)(=O)=O)NC1(CCCC(=O)Nc2cccc(C(C)C)c2)CCC1 57226,C1(C(CNC(C(C)OCOC)=O)(C)C)CCN(C(=O)CC(C)(C)C)CC1 57227,N1(C(C(CCC)F)=O)CCC(C)CC1CNC(c1ccc(OC)nn1)=O 57228,N1(C(C(C)SC(C)C)=O)CCCC2(CNC(c3ccc([N+](=O)[O-])o3)=O)CC12 57229,N1(C(C(CSC)O)=O)CCC12CN(C(=O)CC1(C)CCOCC1)C2 57230,c1(OC(C)=O)c(Cl)cc(NC(=O)CNCCCC23CC(CCO2)C3)cc1Cl 57231,CS(=O)(=O)CCC(=O)NCC(C1CCOC1)NC(c1cocn1)=O 57232,C(N=c1cc(NCC2CC3CCC3C2)nc[nH]1)C1(COC)CCC1 57233,n1(CCC(=O)NCC2N(C(C(C)C(C)(C)C)=O)CCCC2)cnc2ccccc12 57234,CCC(C)CCC(=O)NC(Cn1cccn1)C(=O)N(C1CCCC1C)C 57235,N(C(=NCCC(=O)N1CCCCC1)NCc1cccs1)CC(CC)(CC)N(C)C 57236,c1(CC)cccc(C(N2C(C(=O)NCC3(F)CCCCC3)CCC2C2CC2)=O)n1 57237,C12(C(=O)NCC3CCN(C(C(CC)c4cccnc4)=O)C3)CC(CN1C1CC1)C2 57238,C(=O)(CC(C)(C)CN(C)C)N1CC(OC)C(NC(C2CCCN2C(=O)C(C)C)=O)C1 57239,C1(N(C(C(CC)C)C(=O)O)C2CC2)CCc2nc(-c3ccccc3)ncc2C1 57240,n1(CC(=O)NC(C)CCNC(=O)CC2CCC23CCC3)nc2ccccn2c1=O 57241,Cc1cc(C(=O)NCC2CC(NC(c3ccc(SC(F)(F)F)s3)=O)C2)nc(C)n1 57242,Cc1n[nH]c(C)c1NC(C1CCCN(C(c2cnn(CC3CCCO3)c2)=O)C1)=O 57243,CCCCC(O)C(C)C(=O)NC(C)CN(C)C(c1ncc[nH]c1=O)=O 57244,C1(CC)CN(C(c2cc(OC)cs2)=O)CCC1NC(=O)CCc1ncc(C)[nH]1 57245,n1(C(C(=O)NC(CNC(c2c(CC)n[nH]c2)=O)CC)CC)cnc(C#N)n1 57246,C(=O)(C(C#N)CC)N(CC(=O)NC(C=C)(C)CC)CCC 57247,CC1CC=C(C(=O)N2CC(NC(=O)CCOC3CC3)CC3(CC3)C2)CC1 57248,C1(CNC(CC#N)=O)CCC2(CO1)CC(NC(=O)CCC1CCCCCC1)C2 57249,Cc1[nH]nc2c1CC(C(N1CC(CNC(C3CCCN3N=O)=O)CC1C)=O)CC2 57250,N1(C(C(C)NC(c2ccoc2)=O)=O)CC2(CC(NC(c3cnccn3)=O)CO2)C1 57251,Cn1nc(C(=O)NCCCCCC(=O)NCCc2csnn2)cc1C#N 57252,c1(CC(=O)N(CCCNC(C2ON=C(CC)C2)=O)CC)c[nH]c2cccc(C)c12 57253,C1(NC(C2CN(C)C(=O)C2)=O)CC12CCN(C(c1nccc(C(F)F)n1)=O)CC2 57254,c1(C(=O)NCCCN(C(CC2(COC)CC2)=O)C)cc(C#N)ccc1C 57255,Cc1ccc(Sc2ccccc2C(=O)COC(C2CSCCO2)=O)c(C)c1 57256,N1(C(C2(OC)CCCOC2)=O)CCC(NC(=O)CCn2nc(C)nc2C)C(O)C1 57257,Cc1cc(C(=O)NC2CC(CCNC(=O)COc3ccsn3)C2)c(N)c(F)c1 57258,c1(NC(C(=O)NC(c2csc(C)c2)COC)=O)cnn(C2CCCC2)c1C(F)F 57259,N1(C(CC2CCCC(OC)C2)=O)C2CCC1CC(CNC(c1ccc(Cl)s1)=O)C2 57260,O=C(N=c1[nH]nco1)C12CC(C(=O)NN3CCC(O)CC3)(C1)C2 57261,CN1CCC(CO)(CNC(C23CC2CCN3C(=O)C(O)C2CCCC2)=O)C1 57262,C1(C)(COC)CCCN(C(C2CCN(C(c3cc(C)c(C)[nH]3)=O)CC2)=O)C1 57263,N1(C(C(C)n2cnnn2)=O)CC2CCCC(NC(C34CCC(C3)OC4)=O)C2C1 57264,Cc1cccc2c1OCC2C(=O)NCCOC(C)(C)CNC(=O)CC1CCOC1 57265,C1(C(N2CC3C(N(C(=O)COC4CCC(C)CC4)C)C3C2)=O)(CC)CCOCC1 57266,C12(COC)COC(C(=O)NCC3C=CCN3C(c3cc(C(C)(C)C)n[nH]3)=O)(C1)C2 57267,Cc1cc(NC(=O)CC2C3CN(C(=O)C=Cc4ccc[nH]4)CC23)cc(C)c1F 57268,CCC(CCOC)C(=O)N1CCCCC1CCCNC(=O)C=C1CC1 57269,c1(CC)nc(N2CCC(NC(C3(n4cncn4)CC3)=O)C(F)C2)cc(C)n1 57270,N1(C(c2c(CC)nc(N)s2)=O)CC(C)N(C(=O)CCc2c(C)n[nH]c2C)CC1C 57271,C1(CNC(c2cccc(C3CCOC3)c2)=O)C2CCC(C2)N1C(=O)CC1(O)CCC1 57272,Cc1cc2ccc(C(=O)NC(C)(CNC(=O)CC3(C#N)CCC3)C3CC3)cc2o1 57273,CCC(C)C(=O)C(=O)NCCc1cc(C(N2CCCCC2C(N)=O)=O)no1 57274,C(=O)(CCCC(=O)NC1CCCCC1CNC(C1CC2CCC1C2)=O)OC 57275,c1(C(N(C(C)CC(=O)NCCCCC2CC2C)C)=O)cc(F)ccc1F 57276,C(CCC(C(=O)N1CCCCCCC1)NC(C1CC2CCCC2C1)=O)OC 57277,c1(C(=O)NCCCN(C(c2nc(OC)oc2)=O)C(C)C)c(Cl)oc2ccccc12 57278,C(=O)(C#CC(C)(C)C)NCC(c1ccc(C)cc1)NC(C(CC)OC)=O 57279,c1(C(N(CCCN(C(C(C)C(C)C(C)(C)C)=O)C)C)=O)cc([N+](=O)[O-])ccc1Cl 57280,C1(NC)CN(C(=O)N)CC12CC2.C(C)(C1CC1)=CCO 57281,CC(C)C(F)C(=O)NC1CCN(C(C)C(N2CCCC(C)C2)=O)CC1 57282,c1(C(=O)NC2C(NC(CCC)=O)C2)cccc(N)n1 57283,c1(CNC(C(F)=CC)=O)csc(CNC(c2ccnn2CCF)=O)n1 57284,c1(CNC2CN(C(COC)=O)CC2C)cccc(CNC(=O)OC(C)(C)C)c1 57285,C1(C(N2CCC(COC)(NC(=O)CC(F)(F)F)C2)=O)OC(C)(C)OC1(C)C 57286,CCC(C)CC(C)C(=O)N1CC2CC(C1)N2C(C1(Cl)CC1)=O 57287,CC(C)C(C(=O)N1CCC(CO)C1)C(C)NC(c1nnsc1N)=O 57288,N1(C(C(C(C)C)NC(N)=O)=O)CCCN(C(C2SC3C=CC2CC3)=O)CC1 57289,c1(CNC(C(CSCC)NC(C2CSC2)=O)=O)ccccc1O 57290,Cc1n[nH]c(C)c1CCC(=O)NC1(CNC(c2c(C(C)C)cnn2C)=O)CCC1 57291,CC1(C)COC(C(=O)N(CCNC(c2ccns2)=O)CCOCC2CCC2)C1 57292,C1(NC(C(C=CCCC)O)=O)CCCN(C(c2cc(OC)nc(OC)c2)=O)C1C 57293,c1(N(C)C)ccc(C(=O)NC(C)CCNC(C2CC(OC3CC3)C2)=O)cc1F 57294,c1(C(N2CCCC(C(C)NC(CC=C=C)=O)C2)=O)c(OC)cccc1Cl 57295,CC1=C(C(=O)NCC2CC(NC(c3ccc(Cl)c(Cl)c3)=O)C2)CCCC1 57296,c1(C(N2CCC(CCNC(c3cc(C(N)=O)no3)=O)C2)C)ccccc1Br 57297,C1(NC(C2C(=C)C2)=O)CC2(CCCCN2C(=O)CCc2ccccc2C(N)=O)C1 57298,N1(C(C2CN(S(C)(=O)=O)C2)=O)CCCC(O)(CNC(c2cnc(C(F)F)s2)=O)C1 57299,c1(CC)cn2c(n1)CC(C(N1CC(OCCNC(=O)C(O)C(C)(C)C)C1)=O)CC2 57300,C(C(C(=O)NC1C(O)CC1O)NC(=O)CN(C)C)OCC 57301,c1(CC)oc2ccccc2c1CC(=O)NCC(C)N(C)C(c1ccnc(O)c1)=O 57302,C12(C(=O)NCC3CC(C)N(C(c4ccnc(O)c4)=O)C3)CCCC1CCC2 57303,N1(C(CCC=C)=O)CC2(C1)CN(C(C1CC(S(C)(=O)=O)C1)=O)CC2CO 57304,N(C1COc2cc(Cl)ccc21)C(=O)Nc1cc(C2CC2)ncn1 57305,N1(CC(=O)N(C)C)CCC(C(c2ccccc2)O)CC1.c1(-c2ccccc2)ccncc1 57306,C1(CNC(CCC=CC(C)C)=O)CC2CCC1N2C(c1ccnn1CCF)=O 57307,C(=O)(C(C)C(=O)NC1CCCC(NC(=O)C(C)CO)C1)OC 57308,c1(C(c2n(C(CC)(C)C)nnn2)NC(C)(C)CF)ccc(F)cc1Br 57309,c1(-c2n(C(c3cccc(Br)c3)CC)ccn2)c(C(=O)O)nn2ncccc12 57310,c1(CC)cn2cc(C(N3CCC(N(C(=O)COC(F)(F)F)C)C3)=O)cc(F)c2n1 57311,C1(C(N(C)CC2CCCN2C(c2cc([N+](=O)[O-])n[nH]2)=O)=O)CCCCCC(=O)C1 57312,C1(C(=O)NCC(C)N(C)C(c2csnc2Cl)=O)CCCCC12CCC2 57313,C1(CC(=O)NCC(C2CCN(C(c3cccc(F)c3)=O)CC2)C)COCCOC1 57314,C1(NC(=O)Nc2n(C)nc(C(F)F)c2)CCCC(C(F)F)CC1 57315,CC1(C(=O)NCC2(NC(=O)Cc3cccc(C(F)F)c3)CCC2)CCCCCC1 57316,N1(C(c2sc(C=O)c(Br)c2Br)=O)CCC2(CC1)CC(C(N1CCC(O)C1)=O)CO2 57317,C12(C(N(C(C)CNC(=O)CCC3CC3)C)=O)COC(C(F)(F)F)(C1)C2 57318,C(C(CC(=O)N(C)CC1(F)CCCC1)NC(C1OCCOC1C)=O)OC 57319,C1(NC(c2cc(O)ncn2)=O)C2CCN(C(=O)CCCC3CCCCC3)C12 57320,c1(NC(CCN(C(=O)CCOC2COC2)C)=O)cncc(C(N)=O)c1 57321,C(=O)(C(F)CC(C)(C)NC(c1ccc(N)c(F)n1)=O)N1CC(CN(C)C)C1 57322,C1(F)(CNC(C(=O)NCC)=O)CCC(NC(=O)C=C(C)Cl)C1 57323,N1(C(c2cc(CC)c(F)cc2)=O)CC(C)N(C(=O)CC(F)(F)CC)CC1C 57324,N1(C(=O)CC2CCC(C3CC3)O2)CCN(C(=O)C(O)C2CCCC2)C(C2CC2)C1 57325,C(=O)(C(CCc1ccccc1F)N1CCCC1CC)NCC(=C)C 57326,C=C(C)C(C)(O)C(=O)NC1CCC(NC(c2ccc(CNC(C)=O)cc2)=O)CC1 57327,C1(C(=O)NCCc2c(C)ccc(C)c2)CC2CCCCC2N1C(c1cocn1)=O 57328,C1(C(N2CCCC(CNC(C(C)C3CCCO3)=O)C2)=O)CCCCC12OCCO2 57329,C1(CNC(C2CC(CC)C2)=O)(OC)CCN(C(=O)C(O)Cc2cnn(C)c2)CC1 57330,C1(OC)CC(C(N2CC(C(C)C)C2)=O)N(C(=O)Cc2ccns2)C1 57331,c1(C(=O)NCC(N(C)C(C2(C)C=CCC2)=O)C2CC2)cc2n(n1)CC1(CC1)C2 57332,C(=O)(C(C)(C)S(C)(=O)=O)N1CC(O)(CN(C)C(C2CCC3(CCOC3)O2)=O)C1 57333,N1(C(C(CCCCC)O)=O)CC2(CCCCN2C(C23CC(C)(C2)OC3(C)C)=O)C1 57334,c1(CC(=C)Br)nnc(N2CCC(CCF)CC2)n1CCCc1ccc(OC)cc1 57335,C1(F)(CNC(c2n(C=C)ncc2)=O)CCCN(C(c2ccc(C(F)F)o2)=O)CC1 57336,N1(C(C2(CNC(CC(C)n3cccc3)=O)CC2)=O)CCC(C2(C)CC2)CC1 57337,c1(C(=O)NCC2CCN(C(C3(C)C(C)C3)=O)C2)ccc2oc(O)nc2c1 57338,C=CCCC(C)NC(=O)C(C)=CCNC(=O)CCc1cnn[nH]1 57339,Cc1cc(Br)c(C(=O)Nc2ccc(C)c(C(C)(C)C)c2)cc1Cl 57340,C1(C)C2CC3C(C2NC(=O)C2=CCCCO2)C13.CC(C)(CO)C1(OCC(=O)N)CC1 57341,c1(NC(C23CC2CN(Cc2cnn(C4CC4)c2)C3)=O)cc(F)ccn1 57342,Cc1ccc(O)cc1C(=O)NC(CC1CC1)CC(=O)N1CCC(C(F)(F)F)C1 57343,c1(C(C)C(N2CCC(N(C(=O)CC(F)(F)F)C3CC3)CC2)=O)cccc(C#N)c1 57344,C(=O)(C1CCc2ccccc21)N(CCCNC(c1cc(C(C)C)on1)=O)CC 57345,CCC(C)(CC(=O)Nc1cnn(CC2CCC2)c1)NC(=O)COCC(C)C 57346,c1(C(=O)NCC2CN(C(C#CC(C)C)=O)C(C)CC2)cccc2c1OCCC2 57347,CC1(C)CN(C(=O)CNC(N)=O)C(CNC(C2SCCS2)=O)CO1 57348,C1(O)(C(C)CNC(=O)Cc2cnns2)CCN(Cc2cc(-c3ccoc3)[nH]n2)C1 57349,C1(S(C)(=O)=O)(C(=O)NCC(CC)(C)NC(C2CCN(C)C2C)=O)CCC1 57350,C1(C(=O)NCCCCC=C)CCC2CCC1N2C(c1cnn2c1CCC2)=O 57351,Cc1ccc(NC(c2cocc2C(=O)OC(C)(C)C)=O)cc1O 57352,C(=O)(CCC(=O)N(C(C)CNC(C12CCC(CC1)O2)=O)C)NCC 57353,c1(OC(C)C)ccccc1C(=O)NC(C)CNC(C1CCCN1C(C)C)=O 57354,N1(C(=O)COc2ccc(Cl)c(Cl)c2)CCC2(CC1)CN(C(C1C=CCC1)=O)C2 57355,c1(C(=O)NCC(C)CNC(=O)CC2CC23CC3)c[nH]c(C(N)=O)c1 57356,C1(N(C(=O)CC2CCC2(C)C)CC)CCCN(C(c2cccnc2S)=O)C1 57357,C1(NC(C2CC(C)(C(=O)OC)C2)=O)CCC(NC(c2ccc(=O)oc2)=O)CC1 57358,C(CS(=O)(=O)CCO)NC(CC(C)c1ccccc1)c1nnnn1CC(F)F 57359,C12CCCN(C1)C2=O.C1(NN(C(=O)COC2CCN(C)CC2)C)CCC(CO)CC1 57360,c1(NC(CCN(c2nnnn2C2CC2)C)=O)cccc(Br)c1 57361,C(=O)(CCCC(CC)NC(=O)CCOCC(F)F)NC(CCC)C(C)(C)C 57362,CCC(F)(C(=O)OC)C(=O)N1CCC(O)(CCNC(=O)C(F)=C(C)C2CC2)CC1 57363,N1(C(Cc2c(C)n[nH]c2)=O)CCC2(CCN(C(=O)CNC(C3CC3C)=O)CC2)C1 57364,N1(C(C2CCC(CC)O2)=O)Cc2[nH]nc(C(N3Cc4c[nH]nc4C3)=O)c2C1 57365,C1(C(N(CCc2cn[nH]c2)CC)=O)CCCN(CCOc2ccccc2C)C1 57366,C1(NC(C2CCC(CNC(C3C(C)=CCS3)=O)O2)=O)CC(=O)N(O)C1 57367,N1(C(c2nc(C)oc2)=O)CCCN(C(=O)CCn2ccc3cccnc23)CC1C 57368,C(c1c(Cl)nc2ccccn12)=CC(N1CCCC(F)(CNC(C2C(C)C2)=O)C1)=O 57369,C(CCC(=O)N1CC(OCC(=O)NCC2CC2[N+](=O)[O-])C1)SC 57370,c1(C(=O)NC2CCC(NC(C3C4CCCC34)=O)CC2)cc(O)cc(F)c1 57371,C1(CN(C)C(C2C3CCCCC23)=O)CCCCN1C(=O)CCC1CCOCC1 57372,N1(C(C(CSCC)NC(c2ccco2)=O)=O)CCCN(C)CC1CC 57373,Cc1c(F)ccc(NC(C2(O)CCN(Cc3c(C(F)F)nn(C)c3Cl)C2)=O)c1F 57374,CC1CN(C(c2cnc(O)c(F)c2)=O)CC2(CCN(C(C34CCC(C3)C4)=O)C2)O1 57375,C1(CC(=O)NC2C(CC)N(C(C3CNC(=O)C3)=O)CC2)CCC2(CC1)OCCO2 57376,CC(C)CCC(O)C(=O)N1CCC2(CC2)CC1C=O.C(=O)(N(C)C1CC1)N 57377,c1(COC)cc(C(N2CC(CCCNC(C3CC3OC)=O)(OC)C2)=O)n[nH]1 57378,c1(Cn2c(C(c3cc(F)ccn3)NCC3(C)C(C)(C)C3)nnn2)ccc(F)cc1 57379,N1(C(CC2(OC)CC2)=O)CC=C(C(=O)NC(C23CCC(CO2)C3)C)C1 57380,CC1CC2CN(C(=O)CC#N)CC2N1C(c1cccc(C(=O)OC(C)(C)C)c1)=O 57381,C=C(F)C1(CC(N2CCCCC2CCN(C)C(c2nc(C)c(C)s2)=O)=O)CCC1 57382,CCCCCCCC(F)C(=O)NC1(C2CN(C(C3CC(F)(F)C3)=O)C2)CC1 57383,Cc1cnc(Cl)c(C(=O)N(C)CC2CCCN2C(=O)C(=O)C2CCCC2)c1 57384,c1(NC(C2C(NCc3ncc(C)c(Br)c3)CCCC2)=O)ccc2oncc2c1 57385,C(=O)(CC1=NNC(=O)C1)N(CCC)CCNC(=O)C=Cc1cnc[nH]1 57386,C1(CNC(COCC(=C)C)=O)CN(C(=O)CCOC2CCCC2)C2CC12 57387,C(=O)(CCN(OC)C(=O)c1cccnc1O)N1C(C(CCC)C)CCC1 57388,c1(NC(c2ccc(C)o2)=O)cccc(NC(c2sccc2C2CC2)=O)c1 57389,C(C(C)C(F)C(=O)NC1CCC(N(C)C)C1)NC(c1cnc(C)o1)=O 57390,CCCCC(CN(C)C(C1CCN(C(C2(CCOC)CCC2)=O)CC1)=O)CC 57391,Cc1cccc(C(N2CC(O)(C(C)(C)CNC(=O)C(O)C3CCC3)C2)=O)c1F 57392,N1(C(C2C(C(C)(C)C)C2)=O)CCC2(CC1)CC2NCC=C1CCSCC1 57393,N1(C(=O)NCCC2(C)N=N2)CCNC(=O)C1c1cccc(Br)c1 57394,C1(C(=O)NCC2CCSC2)(CC)CCCN(C(c2cnccc2C)=O)C1 57395,CCCCC(C(=O)NC)NC(=O)C(C)(C)C(C)NC(=O)CC1CC1CC 57396,c1(CC(=O)NCC2N(C(CSCC#C)=O)CCN(C)C2)cccc2c1OCCO2 57397,c1(OC)cncnc1N(CCCNC(=O)CCOCC(F)F)C 57398,C=CCC(CC)C(=O)NCCC1(NC(=O)Cc2csc(-c3ccoc3)n2)CC1 57399,C1(C(=O)OC)CC(C)CN(C(=O)Cn2cc(-c3cc(Br)ccc3OC)nn2)C1 57400,C(CC(O)CNC(c1cn(C2CCC2)nn1)=O)NC(=O)Cc1cscn1 57401,Cc1scc(C(=O)NC2CC3C(NC(=O)Cc4nccn4C)C3C2)c1C 57402,N#CC1CCC(CC(=O)NCC2(F)CC(CNC(c3cc(Cl)sc3Cl)=O)C2)C1 57403,n1(CC(=O)NCCCN(C(C23CCC(C2)C3)=O)CC)nc2n(c1=O)CCOC2 57404,C(c1cn(C)c(=O)n(C)c1=O)=CC(N1CC(NC(c2c(C)ccs2)=O)C(C)C1)=O 57405,c1(CC(C)NC(=O)NCCCC(C)c2ccccc2)cccc(F)c1 57406,C(N=c1[nH]c(=NCCC(C)(C)CO)c2cc(F)cc(F)c2[nH]1)C1CN(C(C)C)C1 57407,c1(C(=O)NC(c2nc(C3CC3)no2)C)cc2n(c1)CCS(=O)(=O)C2 57408,CC(C)(CNC(C1CCC2(CCC2)C1)=O)CC(=O)NC(C)(C)C(C)(C)C 57409,N1(C(C(c2cccc(Cl)c2)C)=O)CC2CCN(C(=O)Cc3cccs3)CC12 57410,CC(C(=O)N1CC(N(C)C(c2coc(C3CCCC3)n2)=O)C(C)(C)C1)S(C)(=O)=O 57411,Cc1nc2scnc(N3CCCC4CN(C(=O)OC(C)(C)C)CCC34)c-2c1C 57412,c1(C(=O)NCC2CCCN(C(CS(CC)=O)=O)C2)cc2c(C)cccc2o1 57413,C(=O)(C(C)S(N)(=O)=O)NCCn1ncc(C(=O)NC(COC(C)C)(C)C)c1 57414,O=C(CN=c1cc[nH]cc1)NC1(C(=O)NCCC2(O)CCOC2)CC(CO)C1 57415,C1(NC(=O)CCc2cnc[nH]2)CCCCCN(C(c2nccc(Cl)c2F)=O)C1 57416,C1(C(N(C)CC2(CNC(c3ccnnc3)=O)CC2)=O)CCC=CCCC1 57417,CC(C)(C)C(O)CC(=O)N1CCC2(CC1)CC2NC(=O)OC(C)(C)C 57418,c1(C(=O)NC(C2CCN(C(c3n[nH]cc3Br)=O)C2)C)cccc(CO)c1 57419,C(=O)(C1CNC(=O)c2ccccc21)N1CCCCC(CNC(C2(C#C)CC2)=O)C1 57420,c1(C(N2CC(CNC(=O)Cc3cnccc3Cl)C3C2C3)=O)cc2n(n1)CCC2 57421,c1(SCC(c2ccccc2)OC)occc1C(N1CC(OC)C1)=O 57422,N1(C(CCC(C)C)=O)CC2(CC(NC(=O)CC3CCOCC3(C)C)CO2)C1 57423,N1(C(COC(C)=O)=O)CCC2(CC1)CC(C)N(C(=O)C=Cc1ccccn1)C2 57424,N1(C2C(C)SCC2)CCN(c2ccccn2)CC1.C12CCN(C1)C(=O)C2 57425,C1(C)(CNC(c2cc(COC)[nH]n2)=O)CCN(C(c2snnc2C)=O)C1 57426,Cc1cc(C(=O)NC(c2cnn(C)c2)C(=O)NCC2C=CCCC2)ns1 57427,C1(OC)CCC12CC(C(=O)NC1CCCC1(C)CN(C(=O)Cc1ccno1)C)C2 57428,N1(C(CCS(N)(=O)=O)=O)CCCCC12CC(NC(=O)C(=Cc1cccnc1)F)C2 57429,c1(CC(=O)NC(CC2CCCC2)C(=O)NCc2cnc(Cl)s2)cncnc1O 57430,N1(C(CCCN(C(CC2(OCC)CC2)=O)C)=O)CC(C(=O)OC)C(C)C1 57431,c1(C(=O)NCCCOCCNC(c2cc(OCC)n[nH]2)=O)cn(C)nc1C 57432,Cc1cc(NC(C2CSCCN2Cc2ccc(Br)cc2O)=O)c(C)cc1Br 57433,N1(C(C2COCCN(C(c3cn(CC=C)nc3)=O)C2)=O)CCCN(C)C(=O)C1 57434,C1(NC(COCc2ncc(C)o2)=O)CN(C(C2CCOCC2)=O)CCC1F 57435,C=CC1(C(=O)NCCOCCCNC(=O)CCS(C)=O)CCOCC1 57436,Cc1c(C(=O)NC2CC(NC(c3cccc(N)n3)=O)C2)cnc2ccccc12 57437,CC#CCC(C(=O)N(CCC(=O)OCC)C)NC(=O)CCc1cn[nH]c1 57438,c1(CC(N2CCC(C)C(NC(c3cnc(O)s3)=O)C2)=O)ccc2cccnc2c1 57439,N1(C(COCC(=O)NC)=O)CCCC2(NC(=O)Cc3c(C)n[nH]c3C)CC2C1 57440,C1(CCNC(C(C)OCCOC)=O)(NC(CCCCOC(C)(C)C)=O)CCCC1 57441,c1(C(C)C)c(F)cc(NCc2ccc(N3CCCC3=O)cc2)cc1F 57442,c1(C(N(C2C(C)CC2)C)=O)coc2c1CN(C(=O)CCc1nccn1C)C2 57443,N1(C(C2CCC(C(N)=O)O2)=O)CCCC2(CCN(C(c3cccnc3F)=O)C2)C1 57444,C(=O)(CCCC(F)(F)CO)N1CCCC(C(C)NC(c2nccc(C)n2)=O)C1 57445,C1(C)(C(=O)NC(C(C)O)CO)CCCN(C(=O)CCC2CC2C)C1 57446,c1(C(N(CCC)CCN(C)C)=O)ccnc(CNC(=O)C(C)C2CCOC2)c1 57447,C1(C(N2CCC(CN(C)C)CC2)=O)C2CCC(C2)N1C(C1CC2COCC2C1)=O 57448,c1(NC)cncc(C(=O)NC2(C3CCCN3C(c3cc(C)cs3)=O)CC2)n1 57449,c1(CC)sc(=N)[nH]c1C(=O)NCCN(C)C(c1cncc(C(F)F)c1)=O 57450,CC12CN(C(=O)Cn3cnc([N+](=O)[O-])c3)CC1CN(C(C1CCS(=O)(=O)C1)=O)C2 57451,c1(C(=O)NCC2CN(C(C3(CO)CCOCC3)=O)C2)cccc2c1CCCCC2 57452,C1(Cn2cc(CCCC)nn2)CCCC(C(=O)N(C(=O)C(F)(F)CC)CC)C1 57453,CC(C(=O)NCCC1CN(C(=O)CCN2CCN(C)CC2)CCCO1)C(C)(F)F 57454,C=C1CC(C(N2CCCC2CC(C)O)=O)(CNC(c2cc(CO)on2)=O)C1 57455,C1(CC)CNC(=O)CN1C(=O)C(C)(C1CC1)N(C)C(c1cc[nH]c(=NC)c1)=O 57456,c1(NC(C2CCN2Cc2cc(O)ncc2Br)=O)ncnc2occc12 57457,CCC(C)CC(=O)N(C1CC(NC(=O)CCOc2ccccc2F)C1)C 57458,c1(C(=O)NC(CCNC(C(CCC)CC)=O)C)ccc([N+](=O)[O-])cc1C(F)(F)F 57459,N1(C(c2ncc[nH]2)=O)CCCC(C2CCN(C(C3(C(F)F)CCC3)=O)C2)C1 57460,CCCCCCC(=O)N(C)CC1CCN(C(C2(C(=O)OC)CC2)=O)CC1 57461,C1(NC(c2cc(C)on2)=O)CN(C(=O)CC2(O)CCCCC2)CC12CCCC2 57462,C(C1CCC(C)CC1)=C(C(N1CCC(N(C(C2CCN(C)C2=O)=O)CC)C1)=O)C 57463,C1(C(N2CCCCCC(NC(CC)=O)C2)=O)COc2cc(OC)ccc2C1 57464,C(=O)(CS(=O)(=O)C(C)C)N1CCN(C(c2snc(C)c2N)=O)C(c2ncc[nH]2)C1 57465,C(=O)(C(C)(CC)C(N)=O)N1C(CNC(c2c(SCC)ccc(Cl)c2)=O)CC=CC1 57466,c1(C(=O)NCCCCCN(C(c2n(CC)ncn2)=O)C(C)C)occ2c1CCC2 57467,N1(C(C2N(C)C(=O)OC2)=O)C2CCC1CN(C(=O)CC1CCOC(C)(C)C1)C2 57468,C1(C(=O)OC)N(C(=O)CCC(C)NC(c2cocn2)=O)CC1(C)C 57469,N1(C(CC(C(C)C)NC(=O)Cn2cncn2)=O)CCN(C)CC(C)C1 57470,CN(C)NC(=O)CCC(=O)N1CCCC1CNC(c1ccccc1SC(F)F)=O 57471,C(=O)(C(C(C)(C)C)N(C1CCC1)C)N1CC(N(C(=O)C(=O)N(C)C)C)C1 57472,C1(C(N(CC(C)O)CCNC(c2cnn[nH]2)=O)=O)CCOC(C)C1 57473,C1(NC(c2cc(Cl)cs2)=O)CCN(C(=O)C=CCn2cncn2)C12CC2 57474,c1(Cc2n(-c3c(C)nccc3)nc(CC3CC(C(F)F)C3)n2)cccc(F)c1Br 57475,N1(C(c2cc(OCC)n[nH]2)=O)CC(NC(=O)C(C2CCCCC2)F)CC1CO 57476,N1(C(CCc2cnc(C)o2)=O)CCCC(CNC(C2CC2(F)F)=O)CC1 57477,c1(CC(=O)N(C2CC(CNC(=O)Cc3ccns3)C2)C)ccc(Cl)cc1 57478,C(=O)(C1Cc2c(Cl)cccc21)NCC1CC2N(C(CC3CN(C)C3)=O)C(CC2)C1 57479,C1(c2nnnn2C2CCCC2)(NCCCC(=O)OCC)CCCC(C=C)C1 57480,CC1CCC(NS(=O)(=O)CC2CCCCO2)C1 57481,N1(C(C2(C(C)C)CCN(C(CCC(CC)=O)=O)C2)=O)CCCC(C2CCC2)C1 57482,c1(OC)ccc(C(=O)NC2CCC(NC(=O)CSc3nccn3C)C2)o1 57483,C1(n2cc(CCCNC(=O)CCOC3CCOC3)nn2)(C(N)=O)CCOCC1 57484,C(CCCC(=O)NCC1CC(CC)C1)NC(CSCC#C)=O 57485,Cn1[nH]c(C(=O)NCCC2CCN(C(=O)COC3COC3)CC2)nc1=O 57486,Nc1ncccc1C(N1CCC(N(C(=O)CC2CS(=O)(=O)C2)CC2CC2)CC1)=O 57487,c1(OCC(N2C3CC(NC(CC4CC(=O)NCC4)=O)(C3)C2)=O)cc(F)cc(Cl)c1 57488,C(=O)(CC(C)(C)c1ccccc1)NCC(Cn1cc(C(C)OCC)nn1)(F)F 57489,C1(F)(C(=O)NCC(CC)(CC)OC)CCCN(C(c2ccc(C)o2)=O)C1 57490,C1(C(C)NC(C2(O)CN(C(=O)CCCNC(=O)CC(C)C)C2)=O)CC2CCC(C1)C2 57491,c1(-c2cccc(NCC(CO)OCC)c2)cccc2nc(C(=O)NCCC)cn12 57492,Cc1cnn(C)c1CC(=O)NCC1OCCC1C(=O)Nc1ccc(OCF)nc1 57493,C1(C(=O)NCC2OCC(C(=O)NCc3c(C(C)C)n[nH]c3)C2)CC(=O)NC(=O)C1 57494,C(c1cc(Br)ccc1OCC)=CC1=CCN(Cc2ccc(CCCC)cc2)CC1 57495,n1(CCC(=O)NC2C(NC(C3ON=C(CC)C3)=O)CCC2)cc(S(N)(=O)=O)cn1 57496,C1(S(N)(=O)=O)(C(=O)NCCC#N)CC1.n12cc(nn1)CNCC(=O)N(C)CCC2 57497,n1(CC(=O)N(CC(C)NC(c2sccc2-n2cccc2)=O)C)cc(CO)nn1 57498,c1(C(=O)NC(C)Cc2cccs2)ccc2nn[nH]c2c1O 57499,C1(CC)C(O)CCN1C(=O)C(C)(C)CC1CC1 57500,c1(CNC(=O)CC2C=CCC2)cn(C2CCN(C(=O)CSc3cccs3)C2)nn1 57501,N1(C(C2C(C)(C)C2(C)C)C(=O)NCCCOC)CCc2ccc(Cl)cc2C1C 57502,C(=O)(CC1=NNC(=O)C1)N(C(C)CNC(c1ccc(CO)c(F)c1)=O)CC 57503,C1(C(=O)NCCCCN(C(c2cn(C3COC3)nn2)=O)CC)CC12CCSCC2 57504,C(=O)(C(CC1CN(C(C23CC(C2)C3)=O)C1)OC)N1CC(C(=O)OCC)C1 57505,O(NC(=O)C(CNC(=O)CCCCCSC)C(C)(C)C)CC(CC)C 57506,N1(C(c2cnnc(Cl)c2)=O)CCN(C(C2CCCC3CCCN23)=O)CC(O)C1 57507,c1(NC(C(N)=O)=O)cncc(C(=O)NCCN2CC3CCC2C3)c1 57508,C=CCC(CNC(c1ccc(CC(C)C)s1)=O)NC(c1csc(C(C)(C)C)n1)=O 57509,c1(C(N2CC(C(=O)NC(c3ccccc3)CO)(SC)C2)=O)cn2ccccc2n1 57510,N1(C(C2N(C(C)=O)CCC2)=O)CCN(C)C(C(N2CC=CCC2)=O)C1 57511,c1(C(N2CCC(NC(CC(C)CF)=O)C2)=O)cn2c(n1)CCC2 57512,C(N=c1nc[nH]cc1C#N)C1CC(NC(c2ccc(C)nc2)=O)C1 57513,C1(C(=O)NCC(C)C)CCCN(C(C)Cc2ccc(C(C)(C)C)cc2)C1 57514,CS(=O)(=NCC(=O)NCCn1cc(CNC=O)nn1)c1ccc(Cl)cc1 57515,N1(C(CCN(C(C2CCC(=O)CC2)=O)C2CC2)=O)CC2(CCC2)CC1CO 57516,c1(OCCNC(c2cnsn2)C)ccccc1F 57517,c1(C(=O)NC(CC)CNC(c2ccc(-c3ncc[nH]3)cc2)=O)cc(=N)[nH]c(Cl)n1 57518,CC1CC2(CO1)CN(C(=O)CC(C1CC1)NC(C1(SC)CC(=O)C1)=O)C2 57519,C=CCC(CNC(C1CC1(C)C(F)(F)F)=O)NC(=O)C=CC(C)(C)C 57520,N1(c2cc(C)[nH]n2)CCCN(C(C23COCC2C3)=O)CC1 57521,N1(C(C#CCNC(c2cc(CC)ncc2)=O)=O)CC2CCC(C1)N2CC 57522,c1(C(=O)NC(CNC(C(CCCC)O)=O)C2CC2)n[nH]c(C(C)C)c1[N+](=O)[O-] 57523,c1(C(=O)NC(CC)C)ccc(CC2(c3ccccc3)CC2)cc1 57524,c1(C(N(CCC(=O)NCC2C(OC)CCC2)C(C)C)=O)csc(C)c1C 57525,c1(CC)cc(C(=O)NC2(CNC(=O)C=CCn3cncn3)CCC2)cc(N)c1 57526,C(=O)(CC1=CCOCC1)N1C(C(=O)NCc2c(CC)nn(C)c2)CC(F)CC1 57527,CC1(C)CCCN(C(=O)Cc2nnc(O)s2)C1CNC(c1cnc(Cl)s1)=O 57528,c1(OC)ccc(C(C)C(=O)N(C(C)CCNC(=O)C(C)(F)F)C)c(C)c1 57529,C1(C(N2CCC(N(CCCOC)CCO)CC2)=O)CCn2cncc2C1 57530,N1(C(C2C(NC(C(C)C(F)(F)F)=O)C=CCC2)=O)Cc2n[nH]cc2C1CO 57531,CN1CCC(CC(C(=O)O)NC(C2CCCC2CF)=O)CC1 57532,C1(NC(c2nc(COCC)sc2)=O)CC2CCC1N2C(c1cn(C)ccc1=O)=O 57533,C#CCCCCC(=O)N1CC(NC(=O)C(CCC)OCC)C(C)(C)C1 57534,N1(C(c2ccc(C(=O)OC)o2)=O)CC2CCC2(CCNC(=O)C=C(C)C)C1 57535,C(=O)(CS(=O)(=O)C1CC1)N(CCCCCNC(c1ncn2c1CCC2)=O)C 57536,c1(CC(=O)NCCC(C)CCO)cc(F)c(Cl)cc1[N+](=O)[O-] 57537,CC1=C(C(=O)NC2CCCC2NC(=O)CC2CC=CCN2C)CCC1 57538,Nc1ccc(C(=O)NCC(C2CC2)NC(C2(O)CC2)=O)cc1OCCO 57539,C1(NC(c2n(C)ncc2)=O)CN(C(=O)CC2CCNC(=O)C2)C2(CCCCC2)C1 57540,S(=O)(=O)(c1ccc2c(c1)N(C(=O)Nc1ccc(S(C)=O)cc1)CCC2)N(C)C 57541,c1(C(=O)NC(CC)CNC(c2ncc(C)cc2C)=O)cccc(S(=O)(=O)CC)c1 57542,N1(c2snc(C(=O)OC)n2)C2CCC1C(CNC(=O)C(c1cscn1)N(C)C)C2 57543,c1(CC(=O)NCC(F)CNC(c2cc(F)n[nH]2)=O)nccc2ccccc12 57544,CC(C)C(C(=O)NCC1(CNC(c2ccccc2)=O)CC12CCC2)N(C)C 57545,C(=O)(C1OCCc2cc(OC)ccc21)NC1C2CC3(C(=O)OC)C(C2)C31 57546,C1(C#CC(=O)NCc2ccc(C(=O)NC(C)CCOC)nc2)(CC)COC1 57547,c1(NC(c2ccccn2)COC)ccc(S(=O)(=O)NCCCC(F)(F)F)c(Cl)c1 57548,c1(NC(COCC)C)ccc(S(=O)(=O)NC2CCC(C)(C)C(CO)C2)cc1Br 57549,C1(C(=O)NCCN(C(CCc2cc(OC)no2)=O)C(C)C)CCCCC12CCC2 57550,Cc1cc(CC(=O)NC2CC(CCNC(=O)C=CCO)C2)cc(C)c1 57551,c1(C(CNC(C(C)CC2CC2)=O)NC(=O)CN(C)C)cccc(Cl)c1Cl 57552,CC1OC(C)C(C(N2CCN(C(=O)CC3(C)CC3(F)Cl)C(CCO)C2)=O)C1C 57553,COn1cnc(C)c1C(=O)NC1COCCN(C(=O)CCCC(C)C)C1 57554,c1(C(=O)NCC2CN(C(c3c(C)nco3)=O)CC2C)cc2cccnc2s1 57555,N1(CC)CCCCC1C(N1CCC(N(C(=O)Cn2[nH]cnc2=N)C)CC1)=O 57556,C(=O)(CC(C)CC(=O)OC)NCC(CC)(C)NC(=O)CN(C)CCO 57557,N1(C(c2cc(C(C)C)[nH]n2)=O)CCCC(NC(C2(C)CCOCC2)=O)C1 57558,N1(C(CC2C(NC(C(C)=C(CC)C)=O)C2)=O)CCC(CN(C)CCOC)C1 57559,CC(F)(F)C(C)(C)CC(=O)C1=CNN=C2C(C(=O)NCCN2CC2CC2)CC1 57560,C1(CNC(C2C(C)CC(=O)CC2)=O)CC2COCC2N1C(=O)C1=NOC(C)C1 57561,NS(=O)(=O)c1ccc(C(N2CCC(F)C(NC(=O)CCc3cscn3)C2)=O)nc1 57562,C(=O)(C(F)(F)C(F)(F)F)NC1(C2N(C(C(C)OC3CCCC3)=O)CCC2)CC1 57563,C(CS(=O)(=O)CC(=O)NC1COCCC1C(=O)NCc1cc(Cl)ccn1)OC 57564,CC(CCCCl)NC(C1(O)CN(C)C1)(C)C 57565,C1(CNC(c2ccc(COC)[nH]2)=O)CCN(C(=O)COCCSC)C12CC2 57566,C1(C(=O)NCC(C(N2CCC(NC(CC)=O)C2)=O)OC)CCC2(CCC2)O1 57567,c1(C(=O)NC2C3CN(C(C(C)(C)CO)=O)CC2C3)csc2c(F)cccc12 57568,N1(C(C2(CC)CN(C(=O)CC3CC=CCC3)C2)=O)CCC(C)(O)CC1 57569,O=C1CCC(CCC(N2CCCC2C2(NC(c3ccncn3)=O)CC2)=O)CN1 57570,N1(C(Cc2c(C)nsc2)=O)CC2CC2(CNC(=O)C(C)n2ccnn2)C1 57571,c1(C(=O)NCC2CC(NC(C3C(=C)C3)=O)C(O)C2)ccn2c(C)cc(C)nc12 57572,C1(CCNC(c2c(C)con2)=O)CN(C(C2CC2(Cl)Cl)=O)CCO1 57573,N1(C(C(C=C)(C)C)=O)CCC(NC(=O)CC2(C)CC2(Cl)Cl)C(F)(F)CC1 57574,N1(C(CS(CC)(=O)=O)=O)CCC2CCN(C(C3(c4ncco4)CCC3)=O)CC12 57575,N1(C(C(C)OC)=O)CCOCC(NC(C2CSCCS2)=O)C1 57576,CC1(C)CCCN(C(c2cccc(C(F)F)c2)=O)C1CNC(=O)C1=CSCCO1 57577,N1(C(CCN(C(Cc2cccc(C#C)c2)=O)C2CC2)=O)CCOCC2(CC2)C1 57578,C1(C(=O)NC2C(NC(c3n[nH]c(C(C)C)c3Br)=O)C2)CCCCCN1C 57579,Cc1cc2[nH]nc(CNC(=O)NC(c3ccc(C#N)cc3)C)c2o1 57580,C(C(C)(O)CC(=O)NCc1c[nH]nc1C(=O)NC1CCCCC1)OC 57581,Cc1cc(=O)c(C(N2CCC(C(=O)NCC34CC(F)(C3)C4)(CO)C2)=O)c[nH]1 57582,c1(-c2c(OC)c(F)ccc2)cccc2sc(C(N3CC(F)(F)CC3OC)=O)cc12 57583,C(=O)(C(CNC(c1cocn1)=O)C(C)(C)C)Nc1c(OC)c(Cl)ccc1 57584,C1(CC)(NC(C2C3CC3CN2C(C2CC(C#N)(OC)C2)=O)=O)CCOCC1 57585,n1(CC)c(C)cc(C(=O)NC2COCCC2NC(=O)C(C)(F)C(=O)OC)c1C 57586,CC1CCN(CC(=O)NCC2CCN(C(=O)CNC(c3ccncc3)=O)C2)C1 57587,Cc1c(Br)noc1C(=O)NCC#CCNC(=O)C(C)OC1CCCCCC1 57588,Cn1nc(C(N2CC(NC(c3cscc3F)=O)CC(O)C2)=O)c(Cl)c1C(F)(F)F 57589,C12(CNC(=O)NCCN3CCOCC3)CC(c3ccccc3)(CO1)C2 57590,CCC(C)CCCC(=O)NCC(CC)(CC)NC(c1cc(C(=O)OCC)no1)=O 57591,Cc1csc(C(N(c2cccc(Br)c2)NCCOCCC2CC2)=O)c1Cl 57592,CCC(CNC(C1(F)CN(C(=O)C(C)CO)C1)=O)C(C)C 57593,c1(NC(=O)NC2CCCC(SC(C)(C)C)C2)ccc(Br)c(F)c1F 57594,C(CC(=O)N(CC(=O)NC(CO)C1(O)CC1)C)SCC 57595,N1(C(C2(SC)CC2)=O)CCC2CC2(C(=O)NCC2CCCC3(CC3)C2)CC1 57596,C1(NC(N)=O)CN(C(=O)Cc2csc(Cl)n2)CC1c1ccccc1 57597,c1(COC)nn(C)c(Cl)c1C(=O)NC(CCNC(=O)C(C)CSC)CC(C)C 57598,N1(C(c2cccc(OC3CCCC3)c2)C(=O)NCCC)CC2CCN(C)CC2C1 57599,C1(C(=O)NCCN(C(C=C(C)CN2CCOCC2)=O)C)CCCN1CC(C)C 57600,C1(C(=O)OC)C2CN(C(C3(NC(c4cc(Cl)n[nH]4)=O)CCSC3)=O)CC12 57601,C(C)(CO)(C(=O)NCCN1CCCC1)NC(c1ccc(C(C)=O)o1)=O 57602,CC1=CCC=CC1C(N1CC(C)(CC(=O)NCC2(N(C)C)COC2)C1)=O 57603,C12CCCCN(C1)C2=O.c1(C(C)=O)ccc(Br)cc1.C1(C(=O)NC)OCC1(C)C 57604,C1(CC)CN(C(c2cnc(OC)c(F)c2)=O)CCC1NC(=O)CC(=O)OC 57605,N1(C(COCCC=C)=O)CC2CCCN(C(c3cc4cccnn4n3)=O)C2C1 57606,C(=O)(C(C(C)C)C(C)C)N(C1CCN(C(=O)C(c2cncn2C)O)C1)CCC 57607,c1(CCC(=O)NCC(c2ccccc2)C)ccc(OC(F)(F)F)cc1 57608,c1(CCN2CCC(CNC(c3c(C(C)C)ccs3)=O)C2)ccnc(F)c1Cl 57609,C1(NC(c2cc(CCNC(c3ccn(C)c3)=O)on2)=O)C2CCCOC12 57610,C1(N(C(c2c(COC)ccs2)=O)C)CCCN(C(c2cc(C#N)on2)=O)C1 57611,C(=O)(C(F)(F)CCn1ccnn1)NCC(C)CN(C)C(c1cc(Cl)cn1C)=O 57612,Cc1cc(C(N2CC3(C2)CN(C(=O)C(C)n2ccnc2)C3)=O)ccc1Br 57613,Cc1nc(C)c(C(C)NC(=O)C(C2CC2)NC(=O)CCC(C)N(C)C)[nH]1 57614,c1(C(N2CC3C(N(C(c4cc(COC)on4)=O)C)C3C2)=O)cc(O)cc(C#N)c1 57615,C1(CNC(C(C)SC(C)C)=O)CC2(CCN(C(=O)C=CC3CCOCC3)CC2)C1 57616,c1(C(N2CCC(C)(NC(C3C(C)CCCC3)=O)C2)=O)cnc2n1CCS2 57617,c1(C(=O)NC23CC(NC(C4(Cl)C(C)(C)C4)=O)(C2)C3)ccc(-n2cncn2)nc1 57618,c1(C(C(=O)NC2(c3cn(CCC=C=C)nn3)CCCC2)O)ccc(F)cc1C 57619,C#CCC(C)(CC)C(=O)NCC1(O)CN(C(c2cnn(C)c2F)=O)C1 57620,C(=O)(C(C(CC)=Cc1cccnc1)N1CCCCC1C1CC1)NCCCC 57621,C(C1=C(C)OCCS1(=O)=O)NC(NC(C1(C)CC=CCC1)C1CCCN1CC)=NC 57622,N1(C(C(C(=C)Cl)(C)C)=O)CCCC(NC(=O)C2=C(Cl)CC2)C(F)C1 57623,N1(C(c2c(C)nn(C)c2)=O)CCCC(O)(CNC(c2cc(C(N)=O)co2)=O)C1 57624,C(=O)(CCCCCN(C)C(C1CCCCS1(=O)=O)=O)NC(C(C)C)Cc1cccs1 57625,N1(C(C(COCC)N=[N+]=[N-])=O)CC2(CC(C(=O)NC(C)CC(C)C(F)F)CO2)C1 57626,c1(N2CCC(C(=O)OC)(COC)C2)ncc(S(C)(=O)=O)cc1Cl 57627,c1(C(N2CCCC(CCNC(C(CCC)OC)=O)CC2)=O)cc(O)c(O)c(O)c1 57628,CC1=C(C(=O)NC2CC(Nc3ncc4ccnc-4[nH]3)C23CCC3)CCS1(=O)=O 57629,C1(NC(C2(CC#C)CCCCC2)=O)CCN(C(=O)CC)CC1CC 57630,c1(CC(N2CCCC2C2(O)CNC2)=O)ccc(Cl)cc1SC1CC1 57631,c1(C(=O)NC2(C)CCN(C(C(COC)(F)F)=O)C2)ccc2nnn(C)c2c1 57632,C(=O)(C(C)CC(=O)NCC(C(C)(C)C)NC(C1CN(C(C)=O)C1)=O)OC 57633,C1(C(=O)NCCC(CCC)O)CN(C)CCN1C(C1CC(N(C)C)C1)=O 57634,O=C1CCCC(C(N2CCC2C(=O)NCC=Cc2ccccc2)=O)C1 57635,N1(CC(=O)N(CCC)C(c2ccccc2Br)=O)CC(C)C(C)C1C 57636,CC1(CNC(C2C3COCC23)=O)COCCN(C(=O)C2=NOC(C(C)(C)C)C2)C1 57637,Cc1cn2c(C(N3CC(CC(C)NC(=O)CC4CCOC4(C)C)C3)=O)cnc2s1 57638,C1(CCNC(C2CCOCC2)=O)CCN(C(=O)CC2CS(=O)(=O)C2)C1 57639,N1(C(COCCC)=O)CCN(C(=O)C(c2cccc([N+](=O)[O-])c2)C)CC(O)C1 57640,C1(C(=O)NC(CN(CC)CC)C)CCC2CCC1N2C(c1cncn(C)c1=O)=O 57641,C1(N(c2c(Br)cnc(C)n2)Cc2cc(C(C)C)ccc2O)CC2CCCC(C1)N2 57642,C1(CNC(c2ccc(CC(C)C)cc2)C)CC2(C1)CC(C#N)C2 57643,c12ccccc1CC(=O)N2.c1(NC(C2C(C(N)=O)C2)=O)ccsc1 57644,C1(NCC(=O)NC(C(C)C)C)CCCCN(C(c2cccnc2)=O)C1 57645,N1(C(CNS(N(C)C)(=O)=O)=O)CCC(C)(C)C(NC(=O)CC2CCC(F)(F)C2)C1 57646,N1(C(C(C)NC=O)=O)CCC(C(=O)NCCC2CC(=O)C2)CC1 57647,c1(C(=O)NCC(=C)CCNC(=O)C=Cc2cnccn2)nncc2c1CCCC2 57648,C1(CCC(=O)NCC(O)CNC(C2(N(C)C)CC2)=O)(C(=O)OC)CCCC1 57649,C1(NC(COc2c(C)cccc2)=O)CCCN(C(C)C(N)=O)CC1 57650,C1(C(N(CCCN(C(=O)CCN2CCCS2(=O)=O)C)C)=O)CNc2ccnn2C1 57651,Cc1cc(C(C)(C)C(N2CC3CC3C2CNC(=O)CC2CC2)=O)ccc1Br 57652,C(=O)(C1c2c[nH]nc2CN1C(=O)C=CCN(C)C)NCCCN(C)C1CC1 57653,C(C)(CNC(=O)COCCC(C)C)(CNC(=O)CCc1nncs1)OC 57654,N1(C(c2c(CC)cno2)=O)CCC(C(CO)NC(=O)C(C)(C)COC)CC1 57655,c1(C(=O)NC2CCC(NC(=O)Cc3ccns3)C2)ccn2ncnc2c1 57656,n1(CCC(=O)NCCC(C)NC(CSCCCC)=O)ncc(=O)c2ccccc12 57657,N1(C(C(CNC(C2(OC)CC(C)C2)=O)N(C)C)=O)CCc2ccc(C#N)cc21 57658,C1(CC)CCN(C(c2csc(=N)[nH]2)=O)C1CNC(C1C2CN(C)CC12)=O 57659,C1(NC(=O)Cc2cscn2)CCC2(CCN(C(=O)C3=CC4(CCOC4)C3)C2)C1 57660,CCC(C)(C)CC(=O)N1CCC(CNC(c2cc(C)c(C(N)=O)cn2)=O)C(C)C1 57661,C1(NC(C(Cc2cn(C)nc2)O)=O)COCCN(C(=O)CN2CSCC2=O)C1 57662,c1(C(=O)NCC(CC)(C)C(=O)NCCn2ccccc2=O)cccc2ccnn12 57663,C(=O)(C(C)(C)c1ncco1)N1CC(CNC(C(C2CCC2)OC)=O)C1 57664,Cc1cc(CC(=O)NC2CN(C(=O)CCc3cncs3)CC2C(F)F)cc(F)c1 57665,C(CCNC(=O)CC1CCCCC1C)(C(C)C)NC(c1cc(C)sc1)=O 57666,C1(COC)(NC(=O)C(n2nccc2C)C)CCN(C(=O)CSS(C)(=O)=O)CC1 57667,C12(C(N)=O)CN(C1)C(=O)CN(C1CCCCC1)C2=O.c1(C(=O)NCC)ccco1 57668,c1(C(N2CCC(n3cc(C(CC)(C)C)nn3)C2)=O)cc(Br)c(Br)cn1 57669,N1(C(C2C(C)(C)CC2)=O)CC(CO)C2(C1)CN(C(=O)C(C)(O)c1ccccc1)C2 57670,N1(C(c2sc(C)c(O)n2)=O)C2CCC1CC(O)(CNC(=O)Cc1ccco1)C2 57671,N1(Cc2ccc(C)cc2Br)C2CCC1CC(NC(c1c(C)ccnc1O)=O)C2 57672,C12(C(=O)NC3(CCO)CN(C(c4ccc(OC)cc4)=O)C3)CCCCC1C2(F)F 57673,CCCCC(C)CCC(=O)NCCCC1(NC(c2ccn(C)c(=O)c2)=O)CC1 57674,c1(CC)sc(C(=O)NC(C)(C)CN(C)C(c2ccccn2)=O)cc1C 57675,C=CC(C)(C)CCNC(C1(OC)CCN(C(=O)COCC(C)(C)C)C1)=O 57676,c1(OCC(=O)N(C(CCNC(C=C(C)Cl)=O)C)C)cc(F)cc(F)c1 57677,c1(C(C)C)ccc(NC(=O)C(C)N(C(=O)C=Cc2ccsc2)C)cc1 57678,N1(C(c2cnc(NC(C)=O)o2)=O)CC2(CC(NC(C3CCCN3C=O)=O)CO2)C1 57679,C12(NC(c3ccoc3)=O)CN(C(c3cnsn3)=O)CC1CS(=O)(=O)C2 57680,N1(C(CC2(OC)CC2)=O)CCN(C(C2CC2(C)C(F)F)=O)C(CC(F)(F)F)C1 57681,c1(C(=O)OC)sc(C(=O)N(C2CCN(C(C3(CCF)CC3)=O)C2)C)cc1N 57682,C1(CC(=O)NC2(N(C(CC3CC(OC)C3)=O)CC3CC3)CCC2)CCN(C)CC1 57683,C1(Nc2cc(C)n(-c3c(C)cccc3)c2C)Cc2ccc(C#N)cc2C1 57684,N1(C(C2CCC(C)(CC)O2)=O)CCCC(C2CCN(C(C3CCNC3=O)=O)C2)C1 57685,CC(C(=O)N1CCCCC1CCN(C)C(C1(F)CCC1)=O)C(F)F 57686,C=CCC(C)(CC)C(=O)NCCN(C)C(c1cccc(OCC(=O)OC)c1)=O 57687,c1(C(=O)NC(CC)CN(C(=O)C(CSC)OC2CCCC2)C)cnncc1OC 57688,N1(C(CCC)=O)CC(COC)CC1(C)CNC(c1c[nH]nc1OCCN(C)C)=O 57689,N1(C(C(C(C)O)N(C)C)=O)CCC2(CC1)CC(NC(c1cncn1C)=O)CCO2 57690,c1(C(C(=O)NC(CCNC(CC2N(CC)CCOC2)=O)C)=O)c(C)nn(C)c1C 57691,c1(OCCC)cccc(CN2CCNCC2C(=O)NCC)c1 57692,C(=O)(C(F)(F)C(F)F)NCC(N1CCN(C(C2CCC(F)C2)=O)CC1)C(F)(F)F 57693,c1(C(N2CCC(O)(CNC(C(CC)CC)=O)C2)=O)cc(C)c(C#N)cn1 57694,c1(COC)cncc(C(=O)N(C2CCCC(N(C(=O)CSCCOC)C)C2)C)c1 57695,C(C1c2ccsc2CCN1C(C1CCc2nc[nH]c2C1)=O)NC(CCP(C)(C)=O)=O 57696,Cc1cnc(F)c(CN(CC(F)(F)F)C(CO)CO)c1 57697,C(=O)(CCCC(C)(F)F)N(C1C(C)CN(C(C2CC(O)(C(F)(F)F)C2)=O)CC1)C 57698,C1(C)(C(=O)NCCC(CNC(c2ccc(CN(C)C)o2)=O)O)CC2CC2C1 57699,C1(N(CCCCCCCC)C)CN(CC2(C(=O)NC(C3CC3=C)=O)CC2)CCC1CO 57700,N1(C(c2ccc(CN(C)C)[nH]2)=O)CCCCC12CC(NC(C1CN(C)C1)=O)C2 57701,c1(C(N(CC(C)N(C)C(C2CCC(N(C)C)CC2)=O)C)=O)ccc(F)cc1F 57702,C#CCC(O)C(=O)N(C)CC1CCCN(C(=O)C(C)NC(=O)OC(C)(C)C)C1 57703,Cc1cc(C(=O)NC2CC(C(C)NC(C3CCC4CC34)=O)C2)ncc1Cl 57704,c1(OCC23OCCC(OC)(C2)C3)nc(C)nc2sc3c(c12)CCC(C)C3 57705,C1(N(CC(N2CCN(C(C)C(=O)NCC(=O)O)CC2)=O)C)C=CS(=O)(=O)C1 57706,C1(C(N2CC(NC(C3(CC=C)CCC3)=O)C2)=O)CC(=O)N(CCC)C1 57707,n1(CC(=O)NCC2CC(NC(c3cc(Cl)c(Cl)[nH]3)=O)C2)cnc2c1CCCC2 57708,C(N=c1[nH]c2c(c(=NCc3cccc(N)c3)[nH]1)CCCC2)C1CC(C)C1 57709,C1(NC(C(C)CC2CC2)=O)C2CC3CN(C(c4ccc(N)cc4O)=O)C1C3C2 57710,N1(C(=O)CN2CCCNC2=O)CCCCC1C1CCCN1C(=O)CSC(F)(F)F 57711,C1(CCNC(C2(CO)CC2)=O)CCN(C(C2CCCC2c2nc(S)n[nH]2)=O)CC1 57712,C(=O)(C(CCN(C)C)NC(=O)C(C)C#N)NC1C(C)CC1 57713,N1(C(C(CC)CC)=O)CC2OCCN(C(C3CCC4CC34)=O)C2C1 57714,c1(CC)c(C(=O)NCC2CC(C)(C)CN2C(=O)C(C)N(C)C(C)=O)cccc1C 57715,C(COC)(CC(=O)N1CCCC1)OC(C(=O)Oc1cccc(C#N)c1)COCC 57716,CS(=O)CCC(O)C(=O)NCCCNC(=O)Cc1cccc(CC(F)(F)F)c1 57717,Cc1ccc(C2CCN(C(=O)CC3CC(NCc4cccnc4Cl)C3)CC2)cc1 57718,N1(C(c2ncc(CC)s2)C(=O)NCCC2CC2)CCCOCC1C 57719,Cc1cc(N(C2CCC2)C)nc(=NCCOc2conc2C)[nH]1 57720,n1(CCC)cccc1C(N1C(C(=O)N(C)CCc2ncccn2)CC1C)=O 57721,CC(C)(CNC(c1occc1C1CC1)=O)CNC(C1(C)CC1Br)=O 57722,N1(C(C2CCC(CNC(C3(C)C(C)C3)=O)O2)=O)CC2CC(C)C2C1 57723,Cn1nccc1C(=O)NC1CC1C(=O)N(C1CCCCC1)CCO 57724,N1(C(C=NOC)=O)CC2=C(C1)CN(C(=O)Cc1ccsc1C)C2 57725,C1(C(N2CC(NC(=O)CSCc3ncc[nH]3)C2)=O)CC2CCC1NC2=O 57726,C1(c2nnnn2C)(NC(c2ccn(C)n2)CC)CCOC2(CCCC2)C1 57727,S(=O)(=O)(c1ccc(-c2ccccn2)s1)NCC1CC(C)NC1 57728,N1(C(C2CCCO2)=O)CCCC(C2CCCN(CC=C3CCCCC3)C2)C1 57729,C1(C)CCCN(C(=O)C=Cc2cccnc2)C1.C(=O)(CCNC(N)=O)N(C)CN 57730,N1(C(c2c(C)[nH]cc2)=O)CCC(O)C(NC(=O)CSc2nnnn2C2CC2)C1 57731,CC1CN(C(c2cscc2C(F)(F)F)=O)CCN1C(=O)CCSc1nnnn1C 57732,CC(C)(C)CC(O)CC(=O)N1CC(O)CC1CC(N1CCNC(=O)CC1)=O 57733,c1(N2CCCC(C)(C)CC2)nc(N2CCCOC(C(C)(C)C)C2)c2ncsc2n1 57734,C1(CNC(C(C(=C)Cl)(C)C)=O)C(C2CC2)CCN1C(=O)CCc1cnc(C)s1 57735,C1(C2(O)CN(C(c3ccc(CO)cn3)=O)C2)(CNC(=O)CC2COCCO2)CC1 57736,N1(C(C(C2(O)CCCC2)(C)C)=O)CC2CCC(NC(c3ccsn3)=O)CC2C1 57737,C12(C(=O)OC3CCC(c4n(C)cnn4)CC3)CCC(=O)N1CC1(CC1)C2 57738,c1(N(C2CCCC2C)C(=O)CCn2cc(Br)ccc2=O)ccc(Br)cc1CNC 57739,C1(CN(C(c2ccon2)=O)CC)CCCN(C(=O)CN2CCC(C)(O)C2)C1 57740,C1(c2cn(C)nc2)CS(=O)(=O)CCN1C(=O)Nc1ccc(I)cc1Br 57741,N1(c2snc(CC)n2)CCC2(CC1)OCCCC2NC(=O)CN(C)CC 57742,c1(CC)cc(C(N2CCC(CNC(=O)C(C)CSC(F)(F)F)C2)=O)c(C)o1 57743,Cc1c(Cl)c(C(=O)NC2CCCN(C(=O)C(c3ccccn3)O)CC2)nn1C 57744,C12(C(N3C(C)(C)C(CNC(=O)CCC[N+](=O)[O-])CC3)=O)CCOC1CCOC2 57745,C12(COC(c3c(C(=O)OC)cncc3)=O)CC(CNC(=O)C(F)(F)F)(CCO1)C2 57746,Cc1cc(O)nc(CNC(C2CCCC2C(C)C)=O)n1 57747,S(=O)(=O)(c1ccc(-c2cccc(C(F)F)c2)cc1)NC1CCC(=O)NC1 57748,O=C(CC1NC(=O)c2ccccc21)NCC1CCN(C(c2coc(O)n2)=O)C1 57749,N1(C(CSCC#C)=O)CCc2ccccc2C(NC(C2CCC(F)C2)=O)C1 57750,CCCC(C)CC(=O)NC12CN(C(c3cccc(OC)c3N)=O)C(COC)(C1)C2 57751,C1(C(=O)NC2C=CCN(C(C(n3cc(C)nc3)(C)C)=O)C2)CC2CCCC2C1 57752,N1(C(C(CC)C(C)O)=O)CCC2(NC(=O)CCCCCO)CCCCCC12 57753,c1(C(C)NC(c2ccc(-n3c(C)cc(C)n3)cc2)=O)nc2ccccc2[nH]1 57754,C1(NC(=O)NCc2cscc2Br)CCc2ccccc2C1 57755,c1(C(C)SCC)nc(CNC2CCCN2S(C)(=O)=O)n(-c2ccnnc2)n1 57756,CCCC(CCC)=CC(=O)N(C1CC(C#N)C1)CC(=O)N(CCOC)CC1CC1 57757,C1(C(N(C(CNC(=O)OC(C)(C)C)C)CC)=O)CCCCC1OC(=O)C(F)(F)F 57758,C1(NC(CSCCC(C)C)=O)CC2(CCN(C(C3CCC(C)S3)=O)CC2)C1 57759,N1(C(C2CC(n3cc(C(C)CC4CCC4)nn3)C2)=O)CCc2ccncc2C1 57760,N1(C(c2csc3nccn23)=O)CCC2(CCCN2C(c2cc(O)cs2)=O)C1 57761,Cc1nnc2n1CCC2(C)C(=O)NCc1ccc2c(c1)OCC(=O)N2 57762,c1(C(c2n(CCC)nnn2)NCCSc2ccsc2)ccccc1Br 57763,c1(C(=O)NCC2CC(NC(c3c(CC)ccs3)=O)C2)ccnc(C)c1 57764,Cc1ccc(Br)c(C(=O)NC2CCCCC2NC(C2CN(C)C2)=O)n1 57765,CN1CC2CC2(CNc2cccc(Oc3ccc(F)cc3F)c2)S1(=O)=O 57766,C(=O)(C(C)(F)C(=O)NCC1CC(O)CN1C(C1(Oc2cnn(C)c2)CC1)=O)OC 57767,C(CCCCCCC(F)(F)F)NC(CCc1c(-n2cc(CN)nn2)cccc1)=O 57768,Cc1ccnc(C(F)(F)C(=O)NCC2CCCN(C(C3CCCN(C)C3)=O)C2)c1 57769,N1(C(C2C(C(C)(C)C)CC2)=O)CCC(N(C(=O)CCCc2ccccn2)CCO)C1 57770,N1(C(c2c(CC)n(CC)nc2)=O)CC2(CCC2)CC1CNC(C1OCC1(C)C)=O 57771,CCCC(C)(O)C(=O)N(CC(C)N(C(=O)Cc1ccco1)C)C 57772,CC#CCC(C(=O)NC1CC2CC(O)C1C2)NC(c1ccnc(C)c1)=O 57773,N1(C(CNC(=O)OC)=O)CCCC1CNC(=O)CCc1cncn1C 57774,C(=O)(C(C(=O)OCC)C(C)(C)C)NC1(C)CCN(C(c2ccn(CC)n2)=O)CC1 57775,CC1CN(CCN(C)C(C2CN(CC(F)F)CC2C)=O)CC(C)O1 57776,c1(C(=O)NC2C(C)CN(C(=O)C3=CCCO3)CC2)cnn2c1CC(C)CC2 57777,C12(C(N3CC(NC(=O)COc4nc(O)nc(O)n4)C3)=O)CCCCC1OCC2 57778,c1(C(=O)NCCCC(C)NC(C(C(C)(C)C)SC)=O)cc([N+](=O)[O-])ccc1C 57779,c1(C(=O)NC2CN(C(=O)Cc3ccoc3)CC2O)cnc2ccccc2c1 57780,Cc1c(C(=O)NCC(F)CNC(=O)C(c2ccn(C)c2)C)cnn1CC(F)F 57781,N#Cc1cc(-c2cc(C(=O)Nc3ccc4c(c3)CCO4)ccn2)ccc1O 57782,C1(C(=O)NCC2(NC(C3C(C)C3)=O)CC2)COC2CC1C2 57783,Cc1ccc2c(=NCC(=O)N=c3cc[nH]cc3)[nH]c(N3CCCC(C)C3)nc2c1 57784,n1(CC)cc(C(N2CCC(C(C)(C)NC(c3cc(C)cn3C)=O)C2)=O)c(C)n1 57785,N1(C(Cc2c(C)cc(Cl)cc2)=O)CC(C)(C)OC2(C1)CN(C(=O)CC(C)F)C2 57786,C(=O)(CC1=CCOCC1)NCC1(CCNC(C2C(C)(C)NC(=O)C2)=O)CC1 57787,N1(C(c2cccc(COC)c2)=O)CCC(C2CCN(C(=O)C=C3CCC3)C2)CC1 57788,C1(NC(c2n(C=C)nnc2)=O)CC2CN(C(c3ccc(F)c(N)c3)=O)CC12 57789,C1(NC(c2csc(S)n2)=O)CCN(C(=O)CCN2CCCS2(=O)=O)CC1 57790,C(=O)(C(F)CC(C)(C)NC(=O)CCn1ccc(C)n1)N1CC(C#C)C(OC)C1 57791,Cc1cccc2cc(C(=O)NCC3CN(C(=O)COCC(F)F)CCC3C)oc12 57792,C(CCCCCC(=O)N1CCC(NC(C2CC(OC(F)(F)F)C2)=O)C(O)C1)SC 57793,c1(COCC(=O)NC2CC(C)(NC(C3C(C)CC3)=O)C2)ccccc1 57794,n1(CC(=O)NC(CC=C)CNC(=O)CN2CC(C)C2)cnc2c(cnn2C)c1=O 57795,CC1(C(=O)NCCC(O)C(=O)NCC(O)C2(Cl)CC2)C=CCCC1 57796,c1(C(N(CCN(C(=O)Cc2cc(C(C)C)no2)CC)CC)=O)cncc(C)n1 57797,CCC(C)C(C(=O)N1CCC=CC1C(=O)NC(C)CN(C)C(C)C)N(C)C 57798,N1(C(c2n[nH]c(C)c2Cl)=O)CC2CCCC(NC(C3CN4CCN3CC4)=O)C2C1 57799,CC(CS(C)=O)C(=O)N1CC(CCNC(=O)CC2=CCCC2)C1 57800,C1(CC(=O)NCC(C)CN2CCCC2)CCCN(C(c2nc[nH]n2)=O)C1 57801,CC1(C)CCc2sc(C(c3nnnn3C3CCOCC3)NCCC3CC3)cc2C1 57802,CC(C)(CNC(c1ccc(-c2ccccc2)cn1)=O)CC(F)F 57803,C(=O)(C1=CCOC1)NCC1(C(N)=O)CN(C(=O)C(c2ccc(Cl)cc2)=O)C1 57804,C1(NC(C2(CSC)CC2)=O)CCC(N(C(=O)CN2CCOCC2)C)C1 57805,C1(C(=O)NCC(C(C)O)C)CCOCCN1C(C1CCC(O)CC1)=O 57806,N1(C(C2CC(C)=C(C)CC2)=O)CC(NC(C2CCCCO2)=O)C2CCCC12 57807,CCCCCCC(C)CC(=O)NC1(COC)CN(C(c2c[nH]nc2[N+](=O)[O-])=O)C1 57808,c1(C(=O)NCC2(NC(C(F)OC)=O)CCC2)cc(-c2cccnc2)[nH]n1 57809,C(=O)(CCCC(=O)NCc1csc(C(N2CCC2)=O)c1)OCC 57810,CC(C)CC(C(=O)NC(CNC(=O)Cc1nccn1C)C1CCC1)n1ccnc1 57811,C(C(C)(C)CC1CN(C(=O)Nc2csc(CC(F)F)n2)C1)NC(CCOCC)=O 57812,C1(NC(C(N2C(=O)CCC2=O)C)=O)CCN(CCc2ccc(F)c(F)c2)CC1F 57813,c1(C2(C(N3CC(C)(NC(c4c(Cl)cn(C)n4)=O)C3)=O)CCC2)ccccc1C#N 57814,C1(OC)CCCC1C(=O)NC(C)CCNC(c1cn(C)cn1)=O 57815,C(C(CO)CC(C)C)NC(C1(CCNC(C(C)=C2CC2)=O)CCC1)=O 57816,N1(C(c2c(CNC(c3nc(CCC)oc3)=O)c[nH]n2)=O)CC(O)CC1CC 57817,c1(OC)cnc(C(=O)NC(C)(CNC(C2CCCC2O)=O)Cn2cccn2)cn1 57818,C1(NC(c2nn[nH]c2Cl)=O)CCCC(CNC(=O)C(C2CCCO2)C2CC2)C1 57819,C(=O)(C1CCCc2cc(C#N)ccc21)N(CCNC(C(CN(CC)CC)F)=O)C 57820,C=CC(C)CN=C(NCC1CCCO1)NCC1(C(C)(F)F)CCOCC1 57821,Cc1c(C(=O)NCC#CCNC(c2[nH]c3ccccc3c2Cl)=O)nc2sccn12 57822,N1(C(c2c(C(C)OC)nn[nH]2)=O)CC2(CC(NC(=O)C(O)C(C)(C)C)CO2)C1 57823,C(CCC(O)CO)N(C(=O)CC1CC1CNC(C1(CO)CCCCO1)=O)C 57824,C1(CNC(C(c2ccc(C)s2)C)=O)CN(C(=O)CCc2cncc(F)c2)CC1C 57825,c1(C(=O)NC2CN(C(c3ccc(C(=O)OC)[nH]3)=O)C3C2C3)ccccc1[N+](=O)[O-] 57826,c1(C(=O)NCCC2N(C(c3c(CC)scn3)=O)CCC2)cc(C)nc2ncnn12 57827,c1(OC)cc(F)c(F)cc1C(=O)NCC(C)NC(C1CC1c1cnn(CC)c1)=O 57828,C1(OC)CN(C)C(C)(C(=O)NC2CCCCC2CNC(c2[nH]cnc2C#N)=O)C1 57829,C#CCC(CCOC)NC(=O)CC(O)CNC(=O)C(C(C)OC)NC(C)=O 57830,CC1Oc2c(C(N3CC4(CCC4NC(=O)COCCF)C3)=O)cccc2NC1=O 57831,C1(C(=O)NCCN(CCCCCC)C(=O)C(c2ccncc2)C)CCS(=O)(=O)C1 57832,C1(CC)CN(C(c2cc(C)sc2C)=O)CCN1C(c1csc(NC=O)n1)=O 57833,c1(C(=O)NCCCN(C(C2(F)CCOC2)=O)C2CC2)ccc(Cl)cc1C(F)(F)F 57834,N(C1CCCOc2c(F)cccc21)C(c1ccc(SC(F)(F)F)c(F)c1)=O 57835,C(=O)(C(O)CCCNC(c1c[nH]c(=NC)s1)=O)N(CC=C)CCOC 57836,c1(OC(C)C)ccc2ccccc2c1CN1CCC1C(=O)Nc1csc(Br)c1 57837,C1(C2CCCC2)(C(N2CC3(CC(NC(C4CCOC4C4CC4)=O)C3)C2)=O)CCC1 57838,CC1(C)CC1(c1cn(CCC(F)(F)Cl)nn1)NCCNC(=O)CNC=O 57839,c1(NC2C3N(C(c4cc(CCC)on4)=O)CC(CC3)C2)ncc(Cl)cc1[N+](=O)[O-] 57840,c12ccc(cn1)C=CC(=O)N2.c1(CSCC(=O)NC2C(C(N)=O)C2)cccs1 57841,N1(C(C2C(=C)C2)=O)CCC(C)C(NC(c2cc(C3(O)COC3)on2)=O)C1C 57842,c1(C(N2CC(NC(C=Cc3nc(C)c(C)[nH]3)=O)(CO)C2)=O)nccc2occc12 57843,N#Cc1cncc(OCC(=O)NCC2CCCCC2c2ccccc2)c1 57844,Cc1cc(C)c(NC(C2CC3CC3N2Cc2cnc(C3CC3)s2)=O)cn1 57845,C1(CC(=O)NC2C(C)CCN(C(=O)C3=CCCCC3)C2)CC2(CCOCC2)CO1 57846,C12(C(N(CCCn3cc(CC(COC)O)nn3)C)=O)CC3CC(C1)CC(C)(C3)C2 57847,c1(CC)ccc(N)c(C(=O)NC23CCC(NC(C4CCCO4)=O)(CC2)C3)c1 57848,N1(CC)CCCC(NC(=O)CC2CC(F)CN2C(=O)CC2(C)CCOC2)C1 57849,N1(C(c2c(C)nc[nH]2)=O)CC(C)CCC1CNC(=O)COc1ccsn1 57850,N1(C(c2c(C)nsc2)=O)CCC(CNC(=O)CC=Cc2ccccc2)C12CCC2 57851,C#CCC(O)C(=O)N1CCC(C(=O)NCc2cnn(CC)c2C2CC2)C1 57852,S(=O)(=O)(c1ccc2c(c1)NCC2)NCc1c(COC)cccc1 57853,N1(C(c2c(C)nns2)=O)CC2C(CNC(c3ccc(CN(C)C)o3)=O)C2C1 57854,C(=O)(C(C(C)(C)C)NC(c1ccn(COC)n1)=O)NC(CCOCC)C 57855,c1(C(N2CCC(S(N)(=O)=O)C2)C(=O)NCC(C)C)noc2c(Cl)cccc12 57856,N1(C(c2csnn2)=O)CC2CC1(C(=O)NCC1CC(C(F)(F)F)C1)C2 57857,c1(C(N2CCC(N(C(C(F)=CC)=O)CC)C2)=O)ccc(S(N)(=O)=O)c(C)c1 57858,CC1ON=C(C(=O)N2CC(CNC(=O)CN3CCCCCCC3=O)C(O)C2)C1C 57859,c1(C(N2CC(C)(C)C(NC(=O)C(F)C(C)(C)O)C2)=O)cccc2c1CNC2=O 57860,CCCCC(C)C(=O)NC(CNC(C1(CSC)CC(F)(F)C1)=O)CC 57861,CCC(C)C(O)C(=O)NCC1CC2CN(C(c3cc(C)cs3)=O)CC12 57862,c1(C(=O)NCC=CCO)cc([N+](=O)[O-])ccc1-n1cnnn1 57863,C(=O)(C1CC=Cc2ccccc21)N1CCC(C)C(NC(C2CC(C)(F)C2)=O)C1 57864,C(CCC(C)C)(C(=O)N(C)Cc1cc(C)cs1)NC(C(C=C)C)=O 57865,N1(C(c2c(CC)onc2C(F)(F)F)=O)CCC(NC(=O)C=NOC)C(F)C1 57866,C(=O)(C(CC(C)C)N(C)C)NCC(CCOC)NC(C1CC2CCC(C1)O2)=O 57867,c1(C(N2C(C(C)NC(C=C(C)Cl)=O)CCC2)=O)cnc(C)cn1 57868,c1(CCCNC(C(C)C2CC2C(F)(F)F)=O)ccc(OC(F)(F)F)cc1 57869,c1(C(N(CCNC(CC(C)OC)=O)C)=O)cc2cc(Cl)sc2[nH]1 57870,C(CCC(C)(C)C(=O)NC1CCn2nnnc2C1)NC(C(COC)C)=O 57871,c1(NC(=O)Nc2ccc(N3CC4CCC3C4)cc2)ccc(C(F)(F)F)c(I)c1 57872,C1(NC(COCC#C)=O)CCCC1(C)CNC(=O)Cn1ccnn1 57873,C(=O)(C(COC)CC(C)C)NC1CC(CNC(C(CC)SC)=O)C1 57874,CC1CC(NC(c2cc3n(n2)CCO3)=O)CCN1C(c1cc[n+]([O-])cc1)=O 57875,c1(OCC)ccccc1OCCNCC1COCC1(C)C 57876,N1(C(C(C)NC(C)(C)C)=O)CCCC1CCCNC(=O)Cn1cc(Br)cn1 57877,C1(NC(C2(SC)CC2)=O)CN(C(=O)CNC(c2ccsc2)=O)CC1C1CC1 57878,C12(NC(c3ccc(C(F)(F)F)cc3F)=O)CCCC1N(C(=O)C=CI)CC2 57879,c1(C(N(C(CNC(c2cc(C)cc(F)c2)=O)C)C)=O)cc(Br)cc(C)c1C 57880,CC(C)CCCOCC(=O)NC1CCC1NC(C12CSCC1C2)=O 57881,c1(N(CC=C)CC)[nH]c(=NC2CC(N3CCC3)C2)nc2scnc12 57882,c1(C(C(=O)NC(CC)(C)C)N(C)C(C2CCCO2)C)ccc(-c2cnn(C)c2)o1 57883,N1(C(C2(CC)CCCCC2)=O)CCCCC(CNC(c2nccc(Cl)c2C)=O)C1 57884,C1(CNC(=O)CCOCC2CCCO2)CCN(C(C2CC(=C(F)F)C2)=O)CC1 57885,C(CN=C(NCC(C)C)N1CCc2ncsc2C1)C1CC(OC)C1 57886,CC1(C)CC(C(=O)NC(C)(C)CCCNC(=O)CCc2nc[nH]n2)=NO1 57887,C1(C(N2CC(OCC(=O)NC3(CC)CC(OC)C3)C2)=O)CC(OC)C1(C)C 57888,C12(NC(CC(=C=C)C)=O)CCCCCC1N(C(C1CC3(C1)CS(=O)(=O)C3)=O)CC2 57889,C1(CCOC)CN(C(C2CCS(=O)CC2)=O)CCN1C(c1n[nH]cc1Cl)=O 57890,c1(C(N2CC(C(C(N3CC(C(=O)NCC)C3)=O)O)C2)=O)csc(C)n1 57891,N#CC1(C(=O)NCC2CC(F)(CNC(=O)Cc3ccsc3Cl)C2)CCC1 57892,c1(C(=O)NCCCCNC(c2ccc3cnnn3c2)=O)ccc2c(c1)CCC2=O 57893,C1(NC(C(CO)OC)=O)CN(C(c2oncc2C)=O)C2CCCC12 57894,c1(C(=O)NCC(C)N(C(CC(C(=C)C)O)=O)C)ccc2c(c1)NCCC2 57895,CCCCC(CC)CC(c1nnnn1CC)NCc1nccn1-c1ccccc1 57896,N1(C(C(CC)CCOC)=O)CC2CC(C1)CN(C(C1OC(C)(C)OC1(C)C)=O)C2 57897,C(=O)(CC(C)C(=O)NCC(C(=O)N1CC=CC1(C)CO)C(C)C)OC 57898,C1(NC(c2c(C)noc2)=O)CN(C(=O)C=C2CCCCC2)C2CCCC12 57899,c1(OC)c[nH]c(C(N2CCN(C)CC2CNC(=O)CC2CCC(=O)N2)=O)cc1=O 57900,Cc1[nH]c(=NC(C)C2COCCO2)sc1S(N)(=O)=O 57901,c1(OCC)oc(C)nc1C(=O)OC1CC=CCC1NC(=O)OC(C)(C)C 57902,CC(CO)(C(F)F)NC(=O)CC1(CNC(=O)C(N)=O)CC1 57903,C1(C(N(CC(C)CNC(=O)CC2(C)CCC2)C)=O)OCCN(C)C1=O 57904,c1(C(=O)NC2(C(=O)NCC(C)CN(C)C)CCCOC2)cc(O)cc(F)c1F 57905,C1(NC(C(CSC)O)=O)CC(NC(=O)C=Cc2ccc(C)s2)C(O)C1 57906,N1(C(CN(C)C(c2cnns2)=O)=O)CCN(C(=O)C(C)(C)CC2CC2)CC1 57907,Cc1ccc2[nH]c(=NCC3CC4(CC(NC(=O)CC5CCC6CC56)C4)C3)sc2n1 57908,C(CC(O)CO)NC(C(c1ccccc1)NC(CCNC(=O)CO)=O)=O 57909,CCC(N=c1cccc(S(=O)(=O)NC(C)(CO)C2CC2)[nH]1)c1cc(C)ccc1C 57910,C(=O)(C(C(C)C)OCC(C)C)NC1(C=C)CCC1 57911,CC12CC1CCN2c1nnc(-c2ccc(Br)s2)o1 57912,N1(C(C(CC=C)C)=O)CCC2(CNC(c3c(F)cc(F)cc3F)=O)CCCCC12 57913,n1(CCC(=O)NC2CC(O)(CNC(C(C3CC3)OC)=O)C2)nc(C)cc1C 57914,CCC(C)(CNC(=O)C(C)OC(C)(C)C)C(=O)N(C)CCOCCO 57915,C(c1ccc(O)cc1)=CC(=O)NCC1CCC(NC(C(C2CCC2)OC)=O)C1 57916,c1(C(=O)NCCCCN(C(C=Cc2ncc(C)[nH]2)=O)C)cnc2ccccc2c1 57917,c1(C(C(=O)O)N(C2CCCN2C2CCNCC2)CC)ccc(C)c(C)c1 57918,C#CC1(C(=O)NCCn2cc(C)cn2)CCN(C(C2COCCO2)=O)C1 57919,N1(C(CC(C)C2CC2)=O)CCCC(C)(NC(c2ccc(CO)cn2)=O)C1 57920,c1(C(=O)NCCN(C)C(C23C4C5C2C2C3C4C52CO)=O)csc2ccccc12 57921,C1(CNC(=O)COCC=Cc2ccccc2)CN(C(=O)Cc2cn[nH]c2)CCO1 57922,N1(C(C(n2cc(-c3ccc(N)c(F)c3)nn2)C)=O)CCCCC(n2ccnn2)C1 57923,N1(C(c2c(C)c(N)ccc2)=O)CCC(C2CCCN(C(c3occc3Br)=O)C2)C1 57924,CC(C(C)(C)O)N(c1nc(C2CCCCC2)cs1)C(C1CC=CCC1)=O 57925,C1(OCC=C)CCN(C(=O)CC2CC(NC(=O)C(F)F)C2)C1 57926,c1(C(=O)NC2C(CNC(C3N(C)C(=O)CCC3)=O)C2)cc(F)c2ccccc2c1 57927,c1(CCC(=O)C(C2C(C(F)(F)F)C2C)C)ccnc(-n2ccc(C3CC3)n2)c1 57928,N1(CC)CCCCC1C(=O)NC1CC(CC(=O)NCC2CC(=O)N(CC)C2)C1 57929,c1(C(N(C)CC2CCCN(C(COCCCC#C)=O)C2)=O)cc(F)c(F)cc1O 57930,N1(C(C2ON=C(CC)C2)=O)CCN(C(c2cc(Cl)no2)=O)CC1C(C)(C)C 57931,N1(C(c2ccc(=N)[nH]c2)=O)CCC(F)(CNC(=O)CC2CNC(=O)C2)CC1 57932,c1(C(=O)NCC(CNC(c2cc(C)c(C)nc2)=O)CO)ccc2cn(C)nc2c1 57933,CC1CN(CCNC(=O)NC2CC=CCC2n2cccn2)CCO1 57934,C(=O)(CN=c1cc[nH]cc1)N1C(CNC(c2ccc(F)c(C)c2C)=O)C(C)CC1 57935,C1(n2cc(CNC(CCC=C)=O)nn2)CCCN(C(c2ccsc2OC)=O)C1 57936,c1(NC(c2cncc(-c3cc(C)cc(F)c3)n2)=O)cc2nc[nH]c2nc1C 57937,c1(C(C)C(N2CCC(c3cn(CCCCC(=O)O)nn3)CC2)=O)cccc(C#N)c1 57938,c1(C(N2C(C(=O)Nc3cc(SC)n[nH]3)CSCC2)=O)cc(Cl)nc(Cl)c1F 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58008,N1(C(C(C)NC(N)=O)=O)CC23CCCC2(C1)CN(C(=O)CC(C)(F)F)C3 58009,C#CCC(O)C(=O)N1C(C(N2CCC2C)=O)CCC1C(C)C 58010,N1(C(C(C2CCN(C(C(C)(C)C3(O)CCC3)=O)C2)F)=O)C2CSCC1C2 58011,n1(CC)c(SCC(CC(C)C)NC(=O)OC(C)(C)C)nc2ccccc12 58012,C1(NC(CC2C(C)CC2)=O)CC2CC(NC(c3cnn(C)c3C(F)F)=O)CC12 58013,N1(C(c2cnc(C(C)C)nc2)=O)CC=C(CNC(C2CC23CCCCC3)=O)CC1 58014,c1(C(C(=O)NCC(c2c(C)cccc2)C)(C)C)ccc([N+](=O)[O-])cc1F 58015,C(=O)(C(C)CC(N)=O)NC1C(NC(c2ccc(CSC)o2)=O)CC1 58016,c1(OC(c2ncoc2C)c2nnnn2C)cncc(N2CCN(CC)CC2)c1 58017,C1(C(=O)NCC(C)NC(C2CC(O)C2)=O)CCCC1O 58018,C1(C(C(=O)NCCC2CC2)N(C)CC2C(CC(C)C)C2)CC(C)CC(C)C1 58019,N1(C(C2(C(=O)OC)CC2)=O)CC2(C1)CN(C(c1nc(C(C)=O)sc1N)=O)C2 58020,n12nc(C)c(c1C)C2C.c1(C(=O)OC)ccc(NC(C)C(=O)N(C)C)cc1 58021,CC1(CNC(C2CCCC(F)(F)C2)=O)CCN(C(c2sccc2C(F)F)=O)CC1 58022,c1(C(N(CCN(C(c2n(CC)ncc2)=O)C(C)C)C)=O)cnnc(Cl)c1 58023,Cc1ccc2c(CC(=O)NC3(C)CCN(C(=O)C4=CCCCO4)C3)coc2c1 58024,CC1(C)C(NC(C2(c3cccs3)CC2)=O)CC1CNC(=O)Cc1nnc(O)s1 58025,Cc1cnccc1CCNC(=O)CC1CCCN(C(c2cnn(C)n2)=O)C1 58026,N1(C(C(CSC)OC)=O)CC2CCC1CN2C(=O)C(C(C)C)N1CCCCC1 58027,N1(C(c2c(Cl)cc(C)s2)=O)CC2(CCC(CNC(C3(O)CCC3)=O)O2)C1 58028,c1(CC)nn[nH]c1C(=O)NCC(C)(C)CNC(c1ccn(CC)n1)=O 58029,c1(C(N2CCC(O)(C(C)(C)C)C2)=O)cc2cc(Cl)ccc2cn1 58030,CCCCCCCC(F)C(=O)OC(c1ccc(C(F)C(F)(F)F)cc1)=O 58031,N1(C(C2C(OCC)C2)=O)CC(CNC(c2cccc(N3CCOCC3)n2)=O)CC1C 58032,C1(NC(c2c(C)n[nH]c2)=O)CN(C(=O)CC2(C)CC(F)(F)C2)CC12CCC2 58033,n1(C(C(=O)NCCCCNC(COCC=C)=O)C)cnc2ccccc12 58034,N1(C(COCC=C)=O)CC(C(=O)NC2(C(C)O)CC2)C2(CCC2)C1 58035,c1(CC)cncc(C(N2CC=CC(C(=O)NC(C3CCC3)C3CC3)C2)=O)c1 58036,c1(NC)cccc(C(=O)NC(C(C)NC(=O)CCCc2cccs2)C(C)C)n1 58037,C(=O)(C(O)C(F)(F)F)N(CC=CC(=O)NC(C#C)CCC)C 58038,CC1(C)COCCC1CNC(C12CC(NC(c3sccc3CO)=O)(C1)C2)=O 58039,c1(C(=O)NCC2CCN(C(c3scnc3C3CC3)=O)C2)csc(CC2CC2)c1 58040,c1(CCC)cccc(C(=O)NC2CCN(C(=O)NC3CC3)CC2)c1 58041,C1(C(=O)NC2(C)COC(C)(C)CO2)(NC(=O)OC(C)(C)C)CCC(F)(F)CC1 58042,N1(C(C2C(CC)N(C)CC2)=O)C2CCC1C(CNC(=O)CCc1ccsc1)C2 58043,C#CCCCCC(=O)N(C)CC1CCCN(C(=O)C(c2cc(Cl)cc(Cl)c2)C)C1 58044,N1(C(C(c2nc(F)ccc2Cl)C)=O)CCC(C2(NC(C3CC=CCC3)=O)CC2)C1 58045,c1(C2C(C(=O)NCC(C)CNC(=O)C(C)c3ccsc3)C2)ccc(F)c(F)c1 58046,Cc1cc(C(=O)NC(C)CC(C)NC(C2(O)CC2)=O)cc(Cl)c1 58047,c1(C(=O)NCC2(C)CCN(C(c3cnco3)=O)C2)ccc2sc(O)nc2c1 58048,CC1c2nnc(C3CCCC3)n2CCN1C(=O)NCC1CC12CCOCC2 58049,n1(C(C)C)ncc(=NC(=O)C(CC2CCOC2)NC(=O)OC(C)(C)C)[nH]1 58050,CC1CCc2c(C(=O)NC3(C)CN(C(C45CCC(F)(CC4)CC5)=O)C3)csc2C1 58051,C1(F)(CNC(=O)C(=O)NCC2CC2)CN(C(c2csc(CO)n2)=O)C1 58052,C1(C(=O)NCC2(OCC)CN(C)C2)CCCN(C(=O)CC2CCOC2=O)C1 58053,c1(C(=O)NCCCNC(CCCC(CC)C)=O)ccc2c(c1)OCCN2 58054,c1(NCC)cccnc1C(=O)NC1CC(C)N(C(=O)CCSC)C1 58055,N#Cc1cc(NC(C23CC2CN(Cc2ccccc2Cl)C3)=O)cc(Br)c1 58056,c1(C(=O)NCC(CNC(C=C(C)C)=O)O)ccc(F)c(C(F)(F)F)n1 58057,CCC(C(=O)N(C)CCn1cc(-c2sccc2C)nn1)C1CCC(=O)N1 58058,N1(CC(C)(C)C)CCC(C(=O)NCC(C2CCCC2)N)CC1 58059,CCCS(=O)(=O)c1ccc(S(=O)(=O)NCC(=O)NCC(C(=O)NC)C(C)O)cc1 58060,O=C(C1COc2ccccc21)NCCOC1CN(C(=O)CC2(O)CC2)C1 58061,N1(C(CC(C=C)(C)O)=O)CCC2CCC(C1)N2C(=O)C(C)OCCOCC 58062,C=C1CC(C(N2CCCCC2c2ccccc2F)=O)N(C(c2ccncc2)=O)C1 58063,COn1cnc(C)c1C(=O)NC(C1CCN(c2ncc(C)c(CSC)n2)CC1)C 58064,C=CC1(CC(=O)NCc2[nH]nnc2CC)CN(C(C2(COC)CC2)=O)C1 58065,C1(C2CCN(C(c3nn(C)cc3N)=O)C2)(NC(C2CC(OC)C2)=O)CC1 58066,C(=O)(C1=CCC(C)(C)CC1)NCC(CC)(C)NC(C1CC1(COC)COC)=O 58067,c1(CCC(N2CCC3CC3(C(=O)NC3CC3)CC2)=O)cc2ccccc2[nH]1 58068,c1(NC(C2CCCN(c3cc(OC)nc(OC)n3)C2)=O)c(Cl)nc(C)nc1Cl 58069,c1(C(=O)NCC2(O)CCN(C(C3CCCCO3)=O)C2)cc(Br)cnc1S 58070,c1(SCC=C)ccccc1C(=O)NCCNC(c1cnn(C)c1CCC)=O 58071,C1(=O)C(C(C)(C)C)N1.c1(CC)nn(C)cc1C(N1CCC(CC)C1C(=O)O)=O 58072,C1(C#CC(=O)NC(c2ccccc2)C(N2CCCC(C(F)F)C2)=O)(CC)COC1 58073,C1(NC(C2CCC(C)(C)O2)=O)CC2(CCN(C(c3cc(Cl)c(N)cc3F)=O)C2)C1 58074,n1(CC(=O)NCCNC(C(c2ccc(F)cc2)(C)N(C)C)=O)ccccc1=O 58075,C1(C(N2CC(C)(COC(C3C=CCC3)=O)C2)=O)(OC(C)(C)C)CCOCC1 58076,C1(NC(c2nnnn2Cc2cccc(F)c2)C(C)C2CC2)CC(=O)N(C(C)C)C1 58077,c1(C(=O)NCC2OCCN(C(C3CCC(C)CC3)=O)C2)c(F)ccc2nc[nH]c12 58078,c1(OC)cccc(C(=O)NC2CN(C(C3(C(F)(F)F)CCC3)=O)CCC2C)c1F 58079,N1(C(c2c(C)cc(-c3ccccc3)s2)=O)CC(C2CN(C(=O)CC(C)(F)F)C2)C1 58080,c1(SC)nc(C(=O)NCC(O)CCNC(=O)C(O)CC2CC2)cs1 58081,N1(C(COC(CC)C)=O)CCC(CNC(=O)Cn2nc(C)nc2C)(COC)C1 58082,Cc1c(N2C(=S)NNC2)cccc1F.C(CCC(C)(C)C)N1CCCC1c1ccccc1Cl 58083,C1(CNC(c2cc(C)n(C)n2)=O)CCCCN(C(c2ccc(CO)cn2)=O)CC1 58084,C12(c3ccn(CC(=O)OC)n3)CCC(CC1)N2C(=O)C(N1CC2CC2C1)C 58085,N1(C(C(=O)Nc2c(C)nn(C(C)C)c2C)=O)CC2CCCOC2C1 58086,c1(C(=O)NC2C(C)CN(C(c3cnc[nH]3)=O)C2)cnc2c(c1)OCCN2 58087,Cc1ncc(C(=O)NCC2CC(NC(=O)CC34CC(C3)C4)C2(C)C)n1C 58088,N1(C(c2c(NC)cncc2)=O)CCN(C(C23CCC2CC3)=O)C(CO)C1 58089,c1(C2CN(C(=O)N(c3ccc([N+](=O)[O-])s3)C3CCC3)C2)cccc2ccccc12 58090,C12(NC(c3cc(C)n(CCO)n3)=O)CCCN(C(=O)C(C)(C)CO)CC1C2 58091,c1(C(N2CC(NC(CCC(CC)OC)=O)C(F)CC2)=O)ccc2c(c1)CCO2 58092,N1(C(C(OC)OC)=O)CCC2(CCC(CNC(C3CC4CCCCC34)=O)O2)CC1 58093,c1(NCC2(C=C)CCC2)ccc(S(=O)(=O)N2CCC(CC)C2C)cc1F 58094,C1(CC)(CC)CCCN(C(=NCCCCC(C)(F)F)NC(C)C)C1 58095,Cc1ccccc1COCC(=O)NC(CNC(C1CCC12CCC2)=O)C(C)C 58096,C1(N(C(C2C(=C)CC2)=O)CCOC)CCN(C(c2nccn2C)=O)CC1 58097,Cc1cc(C#N)nc(NC23CCCC2CN(C(C2(C)C(C)(C)C2(C)C)=O)C3)n1 58098,Cn1ncc2ncc(C(N3CCC4(CCCN4C(C4CC4F)=O)C3)=O)cc12 58099,CCS(=O)(=O)CC(=O)N1CCC(N(C(=O)CCc2ccncn2)CC2CC2)C1 58100,C(C(C)C(F)C(=O)NCCCc1ccco1)NC(C(C)=CCC)=O 58101,Cc1onc(C2CC2)c1C(=O)NCCCCN(C)C(C1CCOC(C)C1)=O 58102,C1(CNC(C(C(C)C)C)=O)CCN(C(c2ccc(-c3cccs3)o2)=O)CC1(F)F 58103,C1(CC(=O)NC)CN(C(=O)C2=CCSC2)CCN1C(=O)C=C(C)C(C)(C)C 58104,C1(N(C(=O)COCc2ccncc2)C)CC2CC1N(C(=O)C(F)=C1CCC1)C2 58105,c1(C(=O)NC(c2ccc(Cl)cc2)c2ccccc2)ccc(F)cc1I 58106,Cc1cc(C(=O)NC2CCN(C(c3ccno3)=O)C(C)C2)c(C)n1C 58107,CN1CCCCC1C(=O)NCC(C)(C)C(=O)NCCCC1(O)CC1 58108,N1(C(C(C=C)(F)F)=O)CC2CCCC(C1)N2C(=O)C=Cc1ccncc1 58109,C#CCCC(O)C(=O)NCC1(CCNC(=O)C(C)Cc2ccccc2Cl)CC1 58110,S(=O)(=O)(c1ccc(NC2CCSC2)cc1Cl)NC(c1c(C)nns1)C 58111,C1(CCNC(=O)COCCF)CCN(C(=O)COc2ccon2)CC1(F)F 58112,N1(C(C)=O)CC2(C1)CN(C(=O)CCN(C(c1cnc(C)n1C)=O)CC1CC1)C2 58113,C1(NC(CC=C(C)C)=O)CC2(CCN(C(C3CC3Br)=O)CC2)C1 58114,C1(C2(NC(C3CC(CCC)C3)=O)CC2)CCN(C(=O)CN2CCOCC2)C1 58115,c1(CN2CCCC(C(=O)NC(CC)C(=O)OC(C)(C)C)C2)nc2ccccc2n1C 58116,c1(C(=O)NC2(C)CCN(C(Cc3c(CC)con3)=O)C2)nn(C)c(Cl)c1Cl 58117,c1(SCC(N2CCN(C3CC3)CC2)=O)ccc([N+](=O)[O-])o1.c12ccccc1SC2 58118,C1(C)(CNC(Cc2cn(CC)nc2)=O)CC(F)(F)CN1c1nc(C2CC2)ns1 58119,Cc1c(NC(=O)C(C)OC(F)F)cc(F)cc1CO 58120,Cc1cc(C(=O)NC(CC(=O)NCC(F)(F)Cl)C2CC2)cnc1O 58121,CCCC(CNC(c1[nH]nnc1C)=O)C(=O)NC1CC12CC(OC)C2 58122,c1(-c2c(C(=O)NC(CC(=O)O)C(=O)O)cn(C)n2)ccc([N+](=O)[O-])cc1 58123,C1(CCC)CN(C(C2CC2C)=O)CCN1C(=O)CNC(=O)C(F)(F)F 58124,c1(C(=O)NCC2CCN(C(CC)=O)CC2C)cc2c(C)nn(C)c2nc1C 58125,C1(C(=O)NCC(C)N(C(Cc2cc(C(C)C)no2)=O)C)CCC([N+](=O)[O-])CC1 58126,N1(CCCCCNC(C(CC)C)=O)CCC(n2cc(-c3ncc(F)cn3)nn2)CC1 58127,C(c1ccc(Cl)s1)=CC(=O)N(C(=O)C(=O)NCC(F)(F)F)C.C1(=O)CO1 58128,C1(NC(CCc2cc(OC)c(F)cc2)=O)CCC(O)CN(C(C2CCCS2)=O)C1 58129,c1(C(N2CCC2c2ccccc2)CSC)ccc(F)cc1F 58130,CCC(C)CC(C(=O)NCC(O)C(=O)OC)NC(c1cnn(C)c(=O)c1)=O 58131,C1(NC(c2ccoc2)=O)CN(C(c2cccc(OCC(F)F)c2)=O)CC1O 58132,C12(C(=O)NCC3(CCNC(=O)C4=NOCC4)CC3)CCCN1CC(O)C2 58133,c1(OC)ccc(NC(=O)NCn2cc(C(=O)NC3CCOC3C)cn2)cc1 58134,C1(N(C(c2ncc(Cl)s2)C(=O)NCC2CCCO2)C)CCN(C(C)(C)C)CC1 58135,C1(NC(CC2(COC)CC2)=O)CCN(C(C2(C)CCC3CC3C2)=O)CC(C)(C)C1 58136,N1(C(CSc2cn(C)nc2)=O)CCC2CCN(C(=O)CC3CC3(C)C)CC12 58137,Cn1ccc2c(C(=O)NCC3CCCCN3C(C3CS(=O)(=O)C3)=O)[nH]cc2c1=O 58138,c1(C(=O)NCC(C(=O)NCCCCC)N(C)C)cc(C)c(C)cn1 58139,N1(C(C2C(C)C2)=O)CC2(C1)C(NC(c1cc3c(ncn3C)[nH]1)=O)CCS2(=O)=O 58140,c1(C(C)C(=O)NCC2CN(C(c3c[nH]c(=N)s3)=O)CC2O)ccc(F)c(F)c1 58141,C1(N(C(CNC(CCC)=O)=O)C)CCCC(NC(=O)CCOC)C1 58142,C(CNC(C)C)(C(=O)O)N(C(CCSCC)=O)C 58143,C1(C(N(C2CN(C(Cc3c(C)nn(C)c3C)=O)C2)C)=O)CC2(C)CCC1(C)O2 58144,C(=O)(C(CC)(CC)CC)NCc1c(C(N2CCC(OCC=C)CC2)=O)scc1 58145,c1(NC(N2CCCC(C#C)(C)C2)=O)ccc(S(=O)(=O)C2CC2)nc1 58146,C=C(Cl)C(C)(C)C(=O)NC1CCC(NC(c2cc(Cl)c[nH]2)=O)CC1 58147,Cc1cc(C(=O)NC2(C)CCN(C(=O)CCN3CCCCCC3)C2)nc(C)n1 58148,C1(NC(c2scc(C)c2Cl)=O)CCC2CCN(C(C3CC3(F)F)=O)C12 58149,c1(C(=O)NCC2CCN(C(=O)C(O)C(F)F)C23CC3)cc(O)cc(F)c1 58150,C12(CNC(c3cnn(C)c3Cl)=O)CC3CC(CC(C3)C1NC(=O)CP(C)(C)=O)C2 58151,CC(CNC(c1ncncc1N)=O)C(F)C(=O)NC(C)CC1CCCCC1 58152,Cc1cc(C(N2CC(CNC(C3CC3c3ccn(C)n3)=O)C2)=O)n(C2CCC2)n1 58153,c1(NC)cccc(C(=O)NC(CCN(C)C)C(=O)NC(CCOC)C(C)C)n1 58154,N1(C(=O)CC2CC3(CCC3)CO2)CC2OCCN(C(c3ns[nH]c3=O)=O)C2C1 58155,c1(C(N2CC(NC(c3sc(CC)c(C)c3)=O)C(F)CC2)=O)c(F)ccc(F)c1O 58156,C=C1CCN(C(c2cn(C)nc2OC)=O)C(C(=O)NCCC(O)CCO)C1 58157,C1(C(=O)NCc2c(C)cnn2C)CC(N=[N+]=[N-])CN1C(c1cc(F)n(C)n1)=O 58158,S(=O)(=O)(c1ccc(O)c([N+](=O)[O-])c1)NS(CCCC(=O)OC)(=O)=O 58159,c1(N(C2CCN(C(c3ccsc3C(F)(F)F)=O)C2)C)cc(F)ncn1 58160,c1(OCC)ccc2c(C(=O)N(CC(=O)OC(C)(C)C)C)c[nH]c2c1 58161,CC#CCCCC(=O)NC1COCC1C(N1CC(OC)CC(C)C1)=O 58162,Cc1cc(C)c(C(=O)NC2CCN(C(=O)CCC(C)NC(N)=O)C2C)o1 58163,CN1CC(NC(C2CSC(C(F)(F)F)C2)=O)CC1=O 58164,c1(NC)cccnc1C(=O)NC(C)CC(C)NC(=O)COC(C)(C)C 58165,C1(O)(CN(C(C=CC(CC)=CC)=O)C)CCN(C(=O)CC2(O)CCC2)C1 58166,N1(C(C)=O)CC2CC2(C(=O)NC2(c3cccnc3)CC2)C1.N12CC(C1)C2=O 58167,c1(C(=O)NC(CNC(c2cc(C(C)C)nn2C)=O)CO)ccc(N)cc1O 58168,c1(NC(C)CN(C(=O)C2=CCSC2)C)ncnc2c1nnn2C1CC1 58169,c1(C(N2CCN(C(CC3C(C)(C)OCCO3)=O)CCC2)=O)cc2c(s1)CCOC2 58170,N1(C(c2cc(C)sc2)=O)CCCOC(CNC(C2CCCN(C)C2)=O)C1 58171,O=S(=O)(c1ccc(=NCC2CCOC(C3CC3)C2)[nH]c1)NCC12CC(CCO1)C2 58172,c1(CC)noc(C)c1NC(=O)Cc1csc(NC(c2ccc(OC(F)(F)F)s2)=O)n1 58173,N1(C(C2C(CCC)C2)=O)CC2(C1)CN(C(c1cc(CC)ccn1)=O)CCO2 58174,C(CC(C)(C)C)(c1n(CC)nnn1)(C1CC1)NCCS(=O)C(C)(C)C 58175,c1(OC)ncc(F)c(N2CC3CC2CN3Cc2ccnc(Cl)c2OC)n1 58176,c1(N2CC(C)(C)C2C2CC2)ccc(C#N)c(CNS(C)(=O)=O)n1 58177,CC12CCC(C(=O)NCC3CCN3C(=O)CCCOc3ccccc3)(CC1)CO2 58178,c1(CN(C)Cc2cc(F)ccc2Br)cc(F)c2c(c1)CCC2 58179,c1(C(N2CCC(NC(C(CC)n3cccn3)=O)C2CC)=O)ccn2nccc2c1 58180,C1(CNc2nccc(C(=O)OC)n2)CC2COCC2N1c1nnc(C(=O)OC)s1 58181,c1(CC)[nH]c(C(=O)NC2CC(CO)N(C(c3sc(F)cc3Cl)=O)C2)nc1Cl 58182,c1(C(N2CC(NC(C(CSC)O)=O)C(C)C2)=O)coc2c(C)cccc12 58183,C1(C(=O)NCC(C)NC(=O)Cc2cnccn2)CC(=O)N(C(C)(C)C)C1 58184,C(c1ccc(F)cc1)=CC(=O)NCC1CC(NC(=O)C2=CCOC2)C1 58185,c1(C(=O)OC)c(C)ccc(NC(=O)NS(=O)(=O)CC2CCOCC2)c1C 58186,Cc1ccc(CC(=O)NC(C)CC2CN(C(=O)C(C)CSC(F)(F)F)C2)cc1F 58187,C(=O)(C1CCCc2nccn21)N1CC(NC(c2ncc(OC)cn2)=O)(CO)C1 58188,c1(C(N(CCCOCCNC(C(C)C(F)F)=O)C)=O)n[nH]c2cccnc12 58189,c1(CC(=O)NCC2(C(=O)NCC(=C)C)CC2)cc(OC)cc(OC)c1 58190,CC1CC(C(N2CC(CC(C)(C)CNC(=O)CC3CCCCC3)C2)=O)C(=O)O1 58191,CCCC(C(=O)N1CC(NC(C2CC(C)CO2)=O)C(C)C1)N(C)C 58192,C1(C(=O)NC2C(C)N(C(C3CCCC3)=O)CCC2)CC2CCCCCCC12 58193,C(=O)(CS(C)(=O)=O)NC(C)C(C)NC(=O)CCC(=O)c1cccs1 58194,c1(NC(C2CCN(C(c3cnc(Br)o3)=O)CC2O)=O)cc(C(F)F)cc(Br)c1 58195,C1(CNC(c2ccncc2F)c2n(CCC)nnn2)OCCOC1(C)C 58196,N1(C(C(C)c2ccco2)=O)CCCC12CCN(C(=O)CCC(C)(C)N(C)C)CC2 58197,N#Cc1cc(Cl)c(C(N2CCC23CN(C(C2(n4cnnn4)CC2)=O)C3)=O)s1 58198,c1(C(=O)NC(CNC(c2cn(CCC=C)nn2)=O)CC)noc2ncccc12 58199,c1(C(=O)NCCCn2nc(C)c([N+](=O)[O-])c2)cccc2ccccc12 58200,C=CC1(NC(C2CC23CCN(C(=O)Cn2nccn2)C3)=O)CCOCC1 58201,N1(C(CC)=O)CCC(C2CCC2)(CNC(C2CCn3c(C)nnc3C2)=O)CC1 58202,N1(C(C(C(C)C)c2scc(C)n2)=O)CCCCC(NC(=O)CC(C)C)C1 58203,C(=O)(CCCCCCCC(=O)N1CCC(N(C(=O)C(F)CC2CC2)C)CC1)OC 58204,c1(C(C)NC(CNC(C=C(C)C(C)(C)C)=O)=O)cccc(F)c1 58205,c1(C(=O)NC(CCOC)CNC(C2CC=CCC2C)=O)c(OC)ccc(Cl)c1F 58206,CC(C)(C)C(O)C(=O)NCC1CCCCN1C(=O)Cc1n[nH]c(=N)s1 58207,c1(C(=O)NC(C2CCN(C(C=CCCC)=O)C2)C)ccc(F)c(CC)c1 58208,N1(c2cccc(C)c2)N=C(C(=O)NC2CC2NC(c2ccns2)=O)CCC1=O 58209,c1(N(CCC)CCNC(c2coc(C)c2)=O)ncccc1[N+](=O)[O-] 58210,C1(CNC(NCC(CCC)Oc2ccco2)=NC)CCCCN1CC(C)C 58211,C(=O)(C(C)(C)CS(N)(=O)=O)N1CCC(N(C(c2coc(C3CC3)n2)=O)CC)CC1 58212,c1(C(=O)NCC(CNC(C(C)=C2CCC2)=O)(C)C)n[nH]c2ccc([N+](=O)[O-])cc12 58213,C12(CNC(=O)Cc3cccnc3Cl)CCC(CC1)N2C(c1cccc(CO)n1)=O 58214,CN1CCOCC1C(=O)NOCC(N1CC2CC2(C2CCO2)C1)=O 58215,C1(C(N2C(C3CCN(C(=O)Cn4cnnn4)C3)CCC2)=O)CC2(CCCO2)C1 58216,N(C(=NCCCF)NCC1(Cl)CCCC1)CC1CCC(=O)N1 58217,c1(CC)ccc(C)c(C(=O)NC2CCN(C(c3c(F)cncc3Cl)=O)CC2C)c1 58218,C1(C(N(C)CC2(C(=O)C3CC3)CC2)=O)CCCN1C1CC1.C12COC(C1)CNC2=O 58219,C1(C(=O)NC2CC(CNC(Cn3c(C(F)F)cc(C)n3)=O)C2)COCCC1(F)F 58220,C(N=c1[nH]c(=NC(C)c2ncc(C)cn2)c2c(ncn2C)[nH]1)C1(OC)CCSC1 58221,S(=O)(=O)(c1c(Br)cccc1[N+](=O)[O-])N1C(C)CC(C(F)(F)F)C1 58222,C1(OC)CCN(C(C2CCOCCN2C(C2CCSCC2)=O)=O)C12CCC2 58223,C12(NC(C(COC)OC)=O)CCCC1N(C(c1cc(C)cc(Br)c1O)=O)CC2 58224,c1(C(=O)NC2CCN(C(C3(C)ON=C(C)C3)=O)C2)ccc2c(ccn2C)c1 58225,c1(N2CCC(N(C(C(C)Cc3cnc[nH]3)=O)C)C2)ncc2c(n1)CCOC2 58226,C1(C(N2CC3C(NC(c4cc(F)ccc4F)=O)C3C2)=O)CC2CCC(C1)C2(F)F 58227,c1(CC(=O)NC(CC)CNC(=O)C(C)OC)cccc(C(F)(F)F)n1 58228,c1(C(=O)Nc2c(C(=O)OC)ccc(OC)c2)ccc2c(c1)N(C)C(=O)C2 58229,C1(C2(O)CN(C(=O)CN3CCCC3C)C2)(CNC(c2ccc(C)cn2)=O)CC1 58230,C=CC(C)C(C)C(=O)N1CCC(CNC(c2cccc(Br)c2N)=O)CC1 58231,N1(C(CCNS(C)(=O)=O)=O)CCN(C(c2ccsc2)=O)C(C2CCC2)C1 58232,c1(OC)ccncc1C(=O)NCCC1(C)CCN(C(=O)CCc2n[nH]c(=N)s2)C1 58233,C1(CNC(C)=O)C2CCC3(CN(CCSCc4cccc(C#N)c4)CC13)O2 58234,c1(OC(C)C)cccc(C(=O)NCC=CCNC(C2CC23CCOC3)=O)n1 58235,CC1(C(=O)NCC2CC(C(=O)NCCn3ncccc3=O)CO2)C=CCCC1 58236,C1(CN(C(=O)COc2cccc(Br)c2)C)CCCN(C(=O)CCCN(C)C)C1 58237,C1(C2C(C)(C)C2C(=O)NC2CN(C(=O)C3CC3)C2)CCN(c2cnccn2)CC1 58238,c1(NC(Cc2c(C)cccc2)=O)cccc(F)c1C(N1CC2CC(C1)O2)=O 58239,C12(C(=O)NCC3CC(F)(CNC(C(CCCC)C)=O)C3)CC3CC(C(=O)N1)C2C3 58240,CC1(C)C(NC(c2cccnc2C(F)F)=O)CCN1C(=O)C(F)C(F)(F)F 58241,C1(C(N(CC(O)C(F)(F)F)C)=O)CC2CCC(C1)N2C(C1CCC=CCC1)=O 58242,CCC(C(=O)NC1(C)CC(NC(c2ccc(N3CCCCC3)nc2)=O)C1)C(C)C 58243,C(=O)(C(CO)C(F)(F)F)NC(CSC)C(=O)NOCCN(C)C 58244,c1(C(=O)NC2CCN(C(CCCSC)=O)C(C)C2)ccc2c(c1)CC(=O)N2 58245,C1(NC(CCOC(C)C)=O)CCN(C(c2cnc(-c3cccs3)o2)=O)CC(O)C1 58246,C1(N(C)C)CC(C(=O)NC(C(=O)NCCN2CCC2)C2CCCC2)C1 58247,c1(C(C(N2CCC(n3ccnc3)C2)C)=O)ccc(F)cc1 58248,n1(CC(N)=O)cc(C(=O)NC2CCCC2NC(C2CCS2(=O)=O)=O)nn1 58249,C1(F)(C(N2CC3(CCN3C(=O)Cc3c(Cl)cccc3Cl)C2)=O)CCCC=C1F 58250,CC(C)CCC(C(=O)NCc1cnn(C2CC2)c1)NC(=O)C(C)NC(N)=O 58251,C(=O)(C(C)(C)S(C)(=O)=O)NCCC(C)N(C)C(c1coc(N(C)C)n1)=O 58252,CS(=O)C1CN(C(=O)COCCNC(c2ccccn2)=O)C1 58253,c1(SC)cccc(C(N2CCC(C(C)NC(=O)C(=O)N(C)C)CC2)=O)c1Cl 58254,N1(C(C2CC(C(=O)OC)C2)=O)CCCCC1CC(=O)NCCN(C)C 58255,CC12CCOC(C(=O)NC3CCN(C(c4scnc4C(C)(C)C)=O)CC3O)(C1)C2 58256,C1(=CC(=O)NC(C2CC(NC(C3CCCC3F)=O)C2)C)CCCCC1 58257,N1(C(C)C)CCC(CC(N2CC(N(C)C(C3C=CC=CC=C3)=O)C(F)C2)=O)CC1 58258,c1(C(=O)NC2CC3CN(C(C#CC(C)(C)O)=O)C2C3)cccn2cncc12 58259,C1(OC)CN(C)C(C)(C(=O)NCC2CN(C(=O)CCc3cccs3)CCC2C)C1 58260,C(=O)(CCCCC(=O)OC)N1CCC(C(=O)Nc2cccc(C#C)c2)C1 58261,Cc1cccc(C(C)NC(c2cccc(Br)c2Cl)C)c1C 58262,N1(C(c2nc(C)n(C)c2)=O)CCC(C)(C)C1CC(N1CCC(N(C)C)C(C)C1)=O 58263,CC(CS(C)(=O)=O)C(=O)NCC1CN(C(=O)Cc2cocn2)CC(C)(C)C1 58264,c1(C(N(CC(CN(C)C(c2ccccn2)=O)O)C)=O)cnc2c(c1)N(C)CCO2 58265,N1(C(C(CC(=C)C)N(C)C)=O)CCC(C(=O)OCC)C(C2CC2)C1 58266,Cc1cccc2c(C(=O)NCC3CCCN(C(C4CC(C)CO4)=O)CC3)cnn12 58267,C=C(C)CC(C(=O)N1CC2CC1C2NC(=O)C(C)OC)NC(C)=O 58268,C1(O)(CNC(CCCC#CC)=O)CCCN(C(=O)CCC(=O)N2CCCC2)CC1 58269,N1(C(C(CCOC)C)=O)CCC(C)(C)C(C(=O)Nc2ccc(F)nc2C)C1 58270,N1(C(=O)NCC2CCC(C)O2)CCN(C2CC2)c2ccccc21 58271,N1(c2nc(N3CCOCC3)nc(N(CC=C)C)n2)CCC(O)C(C)(C)C1 58272,C1(C(N2CCC(C3(C)N=N3)C2)=O)(NC(C2N(C(C)C)CCC2)=O)CCN(C)C1 58273,c1(C(=O)OC)ccncc1NC(=O)NC(Cc1ccco1)C(=O)OC.C1CS1 58274,CCC(C)(C(=O)N1CCC(CN(C(C2COCCC2(F)F)=O)CC)CC1)C(N)=O 58275,c1(CC(Cn2cc(CONC(C3(F)CCCC3)=O)nn2)O)c(F)cccc1F 58276,CC1(N2CCCC2)CCC(c2nc(NCC34CC(CCO3)C4)no2)CC1 58277,C12(CNC(=O)CCc3cnc[nH]3)CC(CO1)N(C(=O)Cn1nnc(C3CC3)n1)C2 58278,c1(CCCNCC2(CC#C)CCOCC2)cc(C(=O)O)ccc1O 58279,c1(C(=O)NC2C(C(=O)Nc3cnc(C)nc3C)CCC2)c(Br)ccc2c1OCO2 58280,N1(C(CCOCC)=O)CCC2(CNC(=O)CC3CCCCO3)CCCC12 58281,CS(=N)(=O)C1CN(C(c2cn(CCNC(=O)CC(Cl)Cl)cn2)=O)C1 58282,c1(C(N2CC3C(CNC(C4C(C(C)C)CCC4)=O)(C3)C2)=O)n[nH]c2c1COCC2 58283,C(=O)(CCC(C)(C)[N+](=O)[O-])NCCCC(C)NC(CCCn1c(C)nc(C)n1)=O 58284,C1(C(=O)NC2(C(=O)NC(C)Cc3cccs3)CC(O)C2)CCC2(CCC2)O1 58285,c1(C(=O)NC(C)CC2CN(C(C3(n4cc(Br)cn4)CC3)=O)C2)cnn(C)c1 58286,Cn1ccn2ncc(C(=O)NC3CC(CNC(c4cccnc4O)=O)C3(C)C)c12 58287,CCC(CCC(=O)N1CCC(C)(C#N)C1)NC(=O)CN1CC2CC2C1 58288,N1(C(Cc2cc(C)[nH]n2)=O)CCC(CCNC(=O)CCSCC(C)C)CC1C 58289,c1(C(=O)NC(CNC(C2C(=C)C2)=O)C2CC2)cc(F)c(OC)c(Cl)c1 58290,CC1CN(C(c2cnc(F)c(Cl)c2)=O)CCC1CNC(C1(C(N)=O)CCC1)=O 58291,C1(CCC(=O)N(C2C3CN(C(C4(C)CCCOC4)=O)CC23)C)CCCCCC1 58292,C1(F)(C(=O)NCC2(F)CC(NC(CN(S(CC)(=O)=O)C)=O)C2)CC2(CCC2)C1 58293,N1(C(c2c(C)occ2)=O)CCC2(C)CN(C(C3C4CC5C(C4)C35)=O)CC12 58294,c1(C(N2C(C)C(NC(c3ncncc3Cl)=O)CC2)=O)cc2n(n1)CCCC2O 58295,N1(C(C2(C(=O)OC)CC2)=O)CCC2(NC(=O)Cc3ccc(Cl)cc3OC)CC2C1 58296,CC1CCC(CNC(=O)Cc2ccc(F)nc2)CN1C(c1cncn1C)=O 58297,C1(CNC(C(C2CCN(C(C(CC)=CCCC)=O)C2)C)=O)CCOC1(C)C 58298,CC1(C)CN(C(C23CCC(CC2)O3)=O)CCC1NC(=O)CCc1cnn[nH]1 58299,CCC(C)CC(C(=O)N(CC(O)COC)C)NC(c1cc(C)nn1CC)=O 58300,c1(C(=O)NC(CC)CNC(C2CC(O)(C(F)(F)F)C2)=O)cc[n+]([O-])cc1 58301,C1(C(C)NC(=O)C(=O)NCCC(N)=O)CCCN1C(=O)C(F)=CC1CC1 58302,c1(C(=O)NCC2(C(C)(C)O)CN(C(CC)=O)C2)cnc2c(Cl)cccn12 58303,N1(C(C2C(C(C)C)C2)=O)CCN(C(=O)Cc2c(Br)cnn2C)C(CCO)C1 58304,c1(N(CC(C)C)C2CC2)nnc(-c2cnn(C)c2)n1Cc1ccccc1F 58305,C12(NC(=O)CCn3cncn3)CCCC1(F)CN(C(C13CCC(F)(CC1)C3)=O)C2 58306,N1(Cc2cc(C)oc2C(F)(F)F)CCOC(CNC(c2nc(C(C)=O)sc2)=O)C1 58307,N1(C(COC2(C)CCOCC2)=O)CC=C(CCNC(C2CCC(=O)O2)=O)CC1 58308,Cc1nc(C(=O)NNC(=O)C(C)C2CCCC2)cn(C)c1=O 58309,c1(C(C(=O)NCCN(C2CCCCC2)C(c2cnc(C)[nH]2)=O)O)ccccc1Cl 58310,C12(C(=O)NC(C)CC3CCN(C(C4(C)CCCC4O)=O)CC3)CCC(CC1)CC2 58311,N1(C(C2CCC(=O)N2)=O)CCCOC(CNc2nccc(CO)n2)C1 58312,C1(NC(CC2(C)OCCO2)=O)C2CN(C(C3CCCN(C(N)=O)C3)=O)CC12 58313,CC(C)C(O)C(C)C(=O)NCCCC(C)CO 58314,C1(CC)CN2CC1C(=O)NCCCCC2=O.C1(CCCNC(N)=O)CCOC1=O 58315,c1(C(C)NC(C2(C)CCN(C(c3ncc(C)nc3)=O)C2)=O)ccc(C#N)cc1 58316,c1(C(=O)NCC#CCNC(C(CC)CCOC)=O)c(Cl)cc(Cl)cc1Cl 58317,C1(NC(c2cc(C)sn2)=O)CCC12CCN(C(c1cc(Cl)c(F)cc1Cl)=O)CC2 58318,CC1=NN(C)C(=O)C1CC(N1C2CCC1C(NC(c1cccc(F)c1Cl)=O)C2)=O 58319,C1(n2cc(C3C(C(=O)OC)C3)nn2)CCCN(C(C2(C3(C)CC3)CC2)=O)C1 58320,c1(C(=O)NC(CNC(C(CC)O)=O)C2CCC2)cc(C)cc([N+](=O)[O-])c1 58321,c12cc[nH]c1C(=O)NC2.C1(C(=O)OC)CC(C(N2CC(N3CC(O)C3)C2)=O)C1 58322,Cc1cncc(C(N2CC(O)(C3CCCN3C(=O)CN3CCN(C)CC3)C2)=O)n1 58323,CCCCCS(=O)(=O)CC(=O)NCC1CN(C)CCN1C(=O)CC1CS(=O)(=O)C1 58324,c1(C(N2CCCC(Br)C2)=O)ccc(NCc2ccncc2Cl)cc1 58325,C1(CC)CN(C(=O)CCCN(C)C(C)=O)CCC1NC(=O)CCCN1CCCC1 58326,N1(C(c2c(SC)c(Br)ccc2)=O)CC(CC(=O)O)OC2(CCOC2)C1 58327,c1(CC(=O)NCC(C)(C2CCC2)NC(C2CCCCS2)=O)cccnc1Cl 58328,C1(C(NOCCOCC)=O)CCCCN(C(=O)CC(C)C)C1 58329,c1(C(=O)NC(C(C)NC(=O)CNC(=O)NC2CCOCC2)CO)cccnc1O 58330,Cc1ccc(O)c(CNC(C2C=CCN(C(C3(C)CC4(CCC4)C3)=O)C2)=O)c1 58331,C12(C(=O)NCC(C3CC3)SC)CC(C)(CN1C(=O)CCn1ccnn1)C2 58332,N1(C(C=CCC)=O)CCC2(CCCC2NC(c2cnn3c2OCC3)=O)CC1 58333,C1(C(N2C(C)CC(NC(C3C(OC)CCC3)=O)C2)=O)Cc2cccnc2C1 58334,C(=O)(CC(O)C(C)C)NC(CC)CC(=O)NCc1nc(C)c(C)s1 58335,N1(C(COCC(C)C)=O)CC2CN(C(c3ccnc4c3CCO4)=O)CC2(C)C1 58336,c1(C(CC(=O)NC2(c3ccc(CCCCCCC)cc3)CC2)O)ccc(O)c(O)c1.C(=O)(O)O 58337,CC1CCC(NC(c2ccc(CO)c(Cl)c2)=O)CN1C(=O)CCC1CCC1 58338,C(=O)(C(F)C(C)(C)O)NCC1N(C(c2nn(C)c(Br)c2)=O)CC(O)C1 58339,[N-]=[N+]=Nc1ccccc1NC(C1CC2CC1C1CNCC21)=O 58340,c1(C(C)C)ncoc1C(=O)NCC1CC(CNC(=O)CC(=O)N(C)C)CO1 58341,Cc1cccc(Cl)c1CC(=O)NCC1CCN1C(=O)C1=C(Cl)CC1 58342,Cn1nc(O)cc1C(=O)OCc1nccn1Cc1ccccn1 58343,Cc1cnc(C(=O)NC2CCC(C(=O)NCc3ccnn3C)C2)cc1C 58344,c1(C(N2CCC3(NC(c4c(C)ocn4)=O)C(C2)C3)=O)cc(=O)n2nccc2[nH]1 58345,N1(C(C(C)=CC)=O)CCN(C(CNC(c2ccsc2)=O)C(F)F)CC1 58346,c1(C(=O)NCC2C(NC(c3coc(Cl)c3)=O)CCC2)ccc(F)c(Br)c1 58347,C1(NC(c2ccc(OC)o2)=O)CCCC(NC(c2ccnc(C(F)F)c2)=O)CC1 58348,Cc1cc(C(=O)NCc2cnn(C)c2)cc(C)c1O 58349,C(=O)(C1=Cc2ccccc2C1C)NCCN1CCCN(C(C(C)OC)=O)CC1 58350,c1(C(N2CCCN(C(C(CC(C)C)OC)=O)C(C)C2)=O)cccc2cnccc12 58351,CC1CCN(C(c2c[nH]nc2C(F)F)=O)CCN1C(=O)CCc1ccccc1F 58352,Cc1ncc(C=CC(=O)NCCNc2cc(F)c(O)c(Cl)c2)c(O)n1.CS(C)=S 58353,N1(C(c2c(CC)cco2)=O)C2CCC1C(C(=O)NCc1nc(C)co1)C2 58354,CC1(C)CC(CNC(=O)C2=CSCS2)CN1C(=O)COc1ccccc1 58355,Cc1cncc(C(=O)NC(C2CC2C(N2CCOC(CN=[N+]=[N-])C2)=O)C)n1 58356,S(=O)(=O)(c1cnc(Cl)nc1)N1C(C(=O)Nc2c(OC)cccc2)CC(O)C1 58357,C1(N(C(c2cnc(CC)s2)=O)C)CN(C(C2CC2C(C)(F)F)=O)CC1(C)C 58358,c1(C(N(C2CCN(C(C3CCCOC3)=O)C2)CC)=O)cc(C)n(C)c(=O)c1 58359,O=C1NCc2cc(C(N3CCOC4(C3)CN(C(C35CCCC3C5)=O)C4)=O)ccc21 58360,c1(OCC)cnc(C(=O)NCC2(O)CN(C(=O)C(S(C)(=O)=O)C3CC3)C2)c(Cl)c1 58361,CCCCC(CC)C(=O)NC1CC(F)(CNC(c2ccc(COC)c(F)c2)=O)C1 58362,c1(NC(CCC)CCc2ccccc2)cc(N(C)Cc2nc(C)cs2)nc(C)n1 58363,C1(O)(CN(C)C(=O)OC(C)(C)C)CCN(C(=O)C(F)CC2CC(F)(F)C2)CC1 58364,C1(NC(CCOCC#C)=O)CC2(CCCN(C(=O)C(CC(C)C)NC(C)=O)C2)C1 58365,C(c1cccs1)=C(C)C(N1CCC(CN(C)C(C2CC2CF)=O)C1)=O 58366,Cc1cc(=NC(C)C2CC(NC(=O)Cn3cnccc3=O)C2)c([N+](=O)[O-])c(C)[nH]1 58367,CCCC(C(=O)NC1(CO)CN(C(c2ccc(N)cc2[N+](=O)[O-])=O)C1)S(N)(=O)=O 58368,C1(C(N(CC(N2CCCC2)=O)C)=O)CC12CCN(C(=O)CCc1cn[nH]c1)CC2 58369,c1(OC)c(F)cc(S(=O)(=O)N(C)CC2CCCC2(C)C)cc1[N+](=O)[O-] 58370,CC1(C)CC(O)(CC(N2CCC(CNC(c3cc(O)ncn3)=O)C2)=O)CO1 58371,C(=O)(C(C(C)C)NC(C)=O)NCCC(=C)CNC(c1cc(C(C)(C)C)oc1C)=O 58372,C1(OCC(N2CCC(=CCC)C2)=O)CCN(C(c2ccccc2O)=O)CC1 58373,CC#CCCC(=O)N(CC(C)NC(c1oc(C)nc1C(F)(F)F)=O)CC 58374,c1(OC)nc(C(=O)OCC(=O)N(C)CC2CCCCC2)sc1C 58375,C12(C(=O)Nc3c(OC)ccc(C)c3)CCCC1CCN2C(C1CCC1C)=O 58376,CCC(CC(C)C)C(=O)NCC1CC2CCC1N2C(=O)CCn1cccn1 58377,c1(OC)ccc(C2CC2)c(C(=O)NCC2(CCNC(=O)C3=CCCS3)CC2)c1 58378,C1(C(=O)OC)CC12CN(C(C13CC1CCN3C(=O)CC1CC=CC1)=O)C2 58379,C12(C(=O)NCC3CN(C(c4n[nH]c(C)c4Cl)=O)CC3(F)F)CCCCN1CCC2 58380,C(CC(C)C)(C(=O)OCC(c1cnn(C)c1)C)Oc1ccc(C)cc1 58381,c1(C(=O)NC(CNC(CCOCC)=O)C2CC2)occc1F 58382,Cn1ccc(=NC(=O)CC(NC2(F)CCC(=O)CC2)NC(=O)OC(C)(C)C)[nH]1 58383,C1(C(N2CC(CC)(CC)C2)=O)CN(C(=O)C=C(C)C(F)F)CC(C)(C)C1 58384,C1(C(=O)NC2CC(NC(=O)NCC3CC=CCC3)C2)CCCCC1N1CCCC1 58385,n1(C(COC)C)nc(-c2ccccc2)nc1CC(C)CC(C)C 58386,C1(F)(CNC(CC2CCC(C)C2)=O)CCN(C(=O)Cc2csc(C(C)C)n2)CC1 58387,c1(C(N(C2CC3CCC(C2)N3C(C2CNC(=O)C2)=O)C)=O)cc(Cl)cc(Cl)c1Cl 58388,c1(C(C)C)ccc(C(=O)NC2C3CN(C(C4CCC(=O)N4C)=O)CC23)cc1 58389,C1(C(=O)NC(CNC(C=C(C)CN2CCOCC2)=O)(C)CO)CCC(F)(F)C1 58390,c1(C(N2CC(F)CC(NC(C=C(CC)C)=O)C2)=O)cccc2nccnc12 58391,C1(C(N2CCC(NC(CCc3nc(=N)[nH][nH]3)=O)(CO)C2)=O)CCn2cnnc2C1 58392,N1(C(CC2N(C(c3n(C)ccc3)=O)CCC2)=O)CCC2(CNC(=O)N2)C1 58393,N1(C(C(COCC)C)=O)CCC2(CCC(CNC(c3ccc(C)n3C)=O)O2)CC1 58394,C1(C)(CNC(CCN(C(c2c(C)scn2)=O)CCO)=O)CCCC1O 58395,Cc1ccc(Cl)cc1NNC(=O)NCC1COc2ccccc2O1 58396,c1(C(=O)NCC(CC)NC(=O)C(C)P(C)(C)=O)cnc2sc(C)nc2c1 58397,C(CCCC(C)NC(c1ccc(C2CCCO2)[nH]1)=O)NC(C1(C)CC(C)C1)=O 58398,c1(CN2CCN(C(c3cc(COC)on3)=O)CC2)cc(Br)c(N)cc1[N+](=O)[O-] 58399,c1(C(=O)NCCCN(C(c2cccc(C)c2C)=O)C(C)C)ccc2nc[nH]c2n1 58400,N1(C(CN(CCC)C)=O)CC2(CC(NC(C3CCCC(F)C3)=O)CO2)C1 58401,C(c1ccc2c(c1)OCCO2)=CC(=O)OC(c1ncc(C)[nH]1)C1CC1 58402,C(CC(C(C)(C)C)NC(=O)CSS(C)(=O)=O)N(C)C(C1CN(C)CCN1C)=O 58403,C1(CNC(C2CC(C)(C)C2)=O)CN(C(C2CCCC2(F)F)=O)CCCO1 58404,Cc1noc(C)c1S(=O)(=O)N(C1CC2CC1CN2)C(C)CO 58405,C(=O)(CCC(CF)CF)N(C(C)CNC(C1CCOC1)=O)C 58406,CC(CC(F)(F)F)C(=O)N1CCCCC(NC(c2snnc2C2CCC2)=O)C1 58407,c1(OC)c(NC(=O)Cc2csc(NC(c3cn(C)cn3)=O)n2)cccc1F 58408,CC(C)CC(O)C(=O)N1CC(CNC(C23CC(C2)C(C)O3)=O)C1 58409,c1(NC(c2nc(-c3cc(C)c(F)nc3)sc2)=O)csc2nccnc12 58410,N1(C(C2CCCOC2)=O)CCC2C(CCCN2C(c2ncoc2Br)=O)C1 58411,C12(NC(c3c(C)noc3)=O)CCC(C(=O)N(C3CC3)CC3CC3)(CC1)C2 58412,c1(N2CCC(C)(COC)C2)nc(N2CCC(C)(CCO)C2)c2ccc(C)cc2n1 58413,c1(C(=O)Nc2cnc(C)s2)cnc2ccc(-c3cccc(F)n3)cc2c1Cl 58414,Cc1ccc([N+](=O)[O-])cc1C(=O)NCC1CN(C(=O)CCOCC(F)F)CC1O 58415,C1(NC(CC(=O)NCC#C)=O)CCN(C2CCN(C(=O)CSC(F)(F)F)C2)CC1 58416,CC1CN(C(c2ccnc(Cl)c2)=O)CC1NC(c1cc(O)no1)=O 58417,N1(C(C(CC)(C)CO)=O)CC2(CC(NC(c3ncccc3Br)=O)CO2)C1 58418,N1(C(COC)=O)CCC(F)(F)C(CNC(c2cnccc2C(C)(C)C)=O)C1 58419,N1(C(CC(=O)NCC#C)=O)CCC(F)(C(N2CCCC(C(C)C)CC2)=O)CC1 58420,C(C(=O)N1CCCCO1)(c1cn(C)nn1)NC(C(OCC)OCC)=O 58421,c1(C(=O)OC)ccc2c(c1)C(=O)N(CCN=c1ccnc(NCC3CC3C)[nH]1)C2 58422,N#Cc1ccc(C(F)(F)F)c(N2CCC(CCC#N)CC2)c1 58423,Cc1c(C(=O)NC(CO)C(=O)NCC(c2cnn(C)c2)C)cccc1C#N 58424,C(C(=O)NNC(=O)C(C)(C)CCCCNC(C1CCC(F)C1)=O)OCCOC 58425,CC(CNC(c1n[nH]c(=N)[nH]1)=O)CC(=O)N(C(C)C(C)(C)O)C 58426,N1(C(c2c(COC)cco2)=O)CCC(C)C1CNC(=O)CCOc1ccccc1 58427,C1(C)(OCC(=O)N(C2CC(NC(c3conc3C3CC3)=O)C2)C)CCOCC1 58428,c1(C(N2CCC(O)C(C)C2)C(=O)NC(C(=O)OC)C)cc(F)cc(F)c1Br 58429,C1(NC(c2c(CC)nns2)=O)CC(CNC(=O)CCc2c[nH]c(=N)[nH]2)C12CCC2 58430,N1(C(COCCC(C)C)=O)CCCCC(NC(=O)CCCC(C)O)C1 58431,N1(C(c2cc(C)n(C)n2)=O)CCC(C)C(NC(c2csc(C3CCCO3)n2)=O)C1 58432,Cc1cc(C(=O)NC2CCN(C(C3CC3C3(C)COC3)=O)C2)cc2c1CCC2 58433,CCC(C(F)(F)F)OC.C1(=O)CCCO1 58434,C(c1cccc(Cl)c1Cl)=CC(=O)NCCC(C)NC(=O)CC1NC(=O)NC1=O 58435,CC(C)C(C)(CNC(c1nscc1Br)=O)NC(C1C=CCC1)=O 58436,c1(C(N2CC3CC(NC(C4(O)CC(C)(C)C4)=O)C3C2)=O)cncc2ccsc12 58437,CC(C)(C)C#CC(=O)N1CC(CNC(C2(C)C=CCCC2)=O)CC1(C)C 58438,c1(OC)ccc2cccnc2c1C(=O)NC1CCC2(CCN(C(C)=O)CC2)C1 58439,N1(C(c2c(CCC)n[nH]c2)=O)CCCCC(C(=O)NCCC(CCC)C2CC2)C1 58440,c1(C(N2C3CC(N4CC(C)C=C(C)C4)C(C3)C2)=O)ccccc1[N+](=O)[O-] 58441,c1(OC)nc(=NCCN(C(=O)C(C)(O)C2CCC2)C)[nH]c(C)c1F 58442,Cn1cnnc1CCCC(=O)NCC1(F)CC(CNC(=O)CC2CCCO2)C1 58443,CC1OC(C)CN(C(c2c(F)cccc2Br)=O)C1C 58444,C1(NC(C(c2n(C)cnc2)O)=O)CCN(C(=O)CCN2CCCC2=O)CC1 58445,N1(C(CC(C)NC(N)=O)=O)CC2(CCC2NC(c2cc(C(F)F)nn2C)=O)C1 58446,CC(O)CCCNC(=O)CCNC(C1(C(C)(F)F)CC1)=O 58447,CC(C)(O)C(F)(F)C(=O)N1CC(C(N)=O)(CNC(C2CCCC(C(F)(F)F)C2)=O)C1 58448,C1(OC(c2c(OCC)ocn2)=O)CCCN(C(c2cnn(C)c2)=O)C1=O 58449,c1(C(=O)NC2C(CC)CN(C(c3cnn(C)c3N)=O)C2)cc(SC)cc(Cl)c1 58450,C1(NC(CCc2cc(C)no2)=O)CC2C1CCN2C(C1CC2CC(=O)C1C2)=O 58451,N1(C(C(=O)NC(Cc2cccc(C)c2)C)=O)CCC2(CCO2)CC1 58452,CCC(F)(F)C(C)(C)C(=O)N1CCN(C(c2ccc(C(C)C)o2)=O)CC1C 58453,C1(C(C)C)CCOCCN1C(=O)COC1(C)CN(C(=O)C(C)Cn2ccnc2)C1 58454,c1(OC)ccc(C(N2CC(CCO)(NC(=O)CC(C)OC)C2)=O)cc1S(C)(=O)=O 58455,CN1CCN(C(=O)C(C)(C)CC2CCC2)CC1CNC(C1Cc2nncn2C1)=O 58456,NS(=O)(=O)c1nc(C(N2CCC(NC(=O)CCF)C(CO)C2)=O)n2ccccc12 58457,CN1C(=O)c2ccccc2C1C(=O)N1CCCCC1CCNC(C1CC1(C)C)=O 58458,CC#CCCCC(=O)NC(C1(C)CN(C(C2CCC(C#N)CC2)C)CCO1)CC 58459,O=C1Cc2ccc(CC(N3CCCC3c3c(F)cccc3Cl)=O)cc2N1 58460,S(=O)(=O)(c1cccc(=NCC(C)c2nccs2)[nH]1)N(C(C=C)C1CC1)C 58461,N1(c2cc(CC)ncn2)CCCC(CO)(NC(=O)C=Cc2ccc(C)o2)C1 58462,C1(NC(C(C)(N(C(=O)CSCC(F)F)C)C2CC2)=O)CCOC(C)(C)C1 58463,c1(C(N(C2CN(C(C(F)OC)=O)C2)C)=O)n[nH]c(C)c1C 58464,N1(C(C)=O)CCCC1C(=O)N(C)CCNC(=O)CCOCC12CC(CO1)C2 58465,N1(C(COCCOC)=O)CC2C3CCC(C2C1)N(C(C1CCC(C)S1)=O)C3 58466,CON1CCC(C(N2CC(NC(C3CCN(C)C(C)C3)=O)CC(F)C2)=O)CC1 58467,C12(NC(C(CSC)OC)=O)CCC(CN(C(c3cc(CO)on3)=O)C1)C2 58468,c1(-c2cc(C(=O)NCC3(O)CN(CC=CC)C3)sn2)ccc(Cl)cc1 58469,N1(CC=C(C)C)CCCC(C(=O)NC(CC2CC2)CO)C1 58470,c1(OC)cc(C(=O)NC2CCCCC2NC(=O)C2=CCC2)c2c(c1)CCO2 58471,c1(N(C(=O)COC(C2CCOC2=O)=O)C)coc2cccc(F)c12 58472,N1(C(C=CC(C)(C)SC)=O)CC=CC(C(=O)N(C)Cc2sccc2C)C1 58473,C(=O)(C(CN(C)C)CC)NC1CN(C(CCOCCC)=O)C1 58474,c1(OC(C)C)cncc(C(=O)NC2(CNC(c3cc(C#N)c[nH]3)=O)CC2)c1 58475,C(C)(CCC(=O)NC1CCC1C(=O)NCC(O)Cn1cccn1)OC 58476,C(=O)(CC(COC)COC)N1CC(O)(C(C(=O)NCCS(CC)(=O)=O)F)C1 58477,n1(C(CC)C)ncc(C(=O)N(CCCN(C)C(c2snnc2C2CC2)=O)C)c1C 58478,N1(C(c2c(OC)nsc2OC)=O)CCC(C)C(NC(C2CSCCS2)=O)C1 58479,CC(C)(CF)C(=O)NC1CCCCC1NC(=O)COCC1(F)CC1 58480,CCC(CN(C)C)CC(=O)NC1CN(C(c2cc(C(C)=O)on2)=O)C(C)(C)C1 58481,c1(C(=O)NC2CC(NC(c3ncncc3Cl)=O)C23CCC3)cccc2sccc12 58482,N1(C(C2CCC(N(C)C)C2)=O)CCC(NC(=O)C#CC2(C(F)(F)F)CC2)C1(C)C 58483,N1(C(C2(C)CS(=O)(=O)C2)=O)CC(CNC(c2ccc(F)s2)=O)C2(CC2)C1 58484,C1(CC)CC(O)CN1C(c1ccc(OCCO)cc1)C(=O)Nc1ccccc1C 58485,N1(C(CC2(NC(C)=O)CC2)=O)CC2CCN(C(=O)CC3NC(=O)NC3=O)C(C2)C1 58486,c1(C(=O)NC2C(C)CN(C(C3(C)CCC3)=O)CC2)cnc2[nH]ccc2n1 58487,N1(C(CC(C)(C)C)=O)C2CCC1C1CC1(NC(C1CC3CCC1O3)=O)C2 58488,C1(CN(C)CC)CN(C(=O)C(C(C)C)OC2CCCC2)CC(C)(C)C1 58489,C1(C(N2CCC(O)(C(C)NC(C3CC3(F)F)=O)C2)=O)CC(C2CC2)=NO1 58490,C=CC(CCC)CC(=O)N1CC(OCCC(=O)OCC(=O)N(C)C2CC2)C1 58491,C1(C(N(C)CC2(CO)CCC2)=O)(NC(=O)Cc2csnn2)CC(F)(F)C1 58492,C(=O)(C#CC1(C)CC1)NCC1(OC)CCN(C(c2ccc(CN(C)C)o2)=O)C1 58493,Cc1cc(C(=O)N(CCCNC(C2CC3(CCCO3)C2)=O)C2CC2)c(N)c(F)c1 58494,Cc1cnc(C(=O)N(C2CCN(C(=O)CC34COC(CF)(C3)C4)C2)C)cc1C 58495,c1(C(N(C)CC2N(C(C=CC=CC)=O)CCC2)=O)cccn2ncnc12 58496,C1(C(N2CC(CCC#C)C2)=O)CC(NC(=O)Cn2ncnn2)CCO1 58497,C(=O)(C(C(C)C)C(C)C)NC1CC(CNC(C(C(C)(C)C)NC(C)=O)=O)C1 58498,c1(CO)ccc(NCC2(c3cccc(Cl)c3)CCC2)c([N+](=O)[O-])c1 58499,c1(-c2c(C)csc2)cc(C(N2CCC(c3ncccn3)CC2)=O)cc2[nH]ncc12 58500,N1(C(C=CCN(C)C)=O)CCC2(CC1)CN(C(c1cc3c([nH]1)CCCC3)=O)C2 58501,CN=c1nc(C(N2CCCC(O)(CNC(C3CC3Br)=O)C2)=O)cc(C)[nH]1 58502,c1(C(=O)NCC(C2CCOC2)NC(c2sccc2F)=O)c(F)cccc1[N+](=O)[O-] 58503,C1(C(N(C)CC2CC(=C)C2)=O)CC2CCC1N2C(=O)Cn1nnc(C)n1 58504,c1(C(=O)NC(C)CN(C)C(c2ncc(F)cc2F)=O)cc(F)cc(Br)c1F 58505,c1(C(=O)OC(C)Cc2ccco2)cc(Br)c(F)cn1 58506,C(=O)(CS(=O)(=O)CC(=O)NCC1CC(O)CN1C(=O)C(c1ccc(C)s1)C)OC 58507,C1(CN(C2CC=CC2)CCC2(CS(C)(=O)=O)CC2)CCN(C(N)=O)C1 58508,C1(NC(C(N2CCCCCC2)C)=O)CCN(c2ccncc2C#N)CC1O 58509,C1(C)(C(=O)NC(COCC)C(C)C)CCN(C(c2cnc(N)cn2)=O)CC1 58510,C1(C(=O)NC(CNC(CC(CC)C2CCC2)=O)(C)C2CCC2)CC(=O)NC(=O)C1 58511,Cc1cc(O)ccc1CC(=O)NCC1COC(CNC(C2CC(C)(C)CO2)=O)C1 58512,c1(CC)nn(C)c(Cl)c1C(N1CC(CNC(=O)C(C)(O)C2CCC2)C(C)(C)C1)=O 58513,CCCCCCC(CC)NC(C1CC(CCNC(=O)CC(C)n2cccc2)C1)=O 58514,Cc1cc(C(N2CCC(C3CC3)C2CNC(=O)CC(C)(C)O)=O)cc2nc[nH]c12 58515,C=CCCC(C(=O)N(CC(=O)NC)CC)NC(c1ccc(C)cn1)=O 58516,N1(CC(CNC(c2cc(C)sc2)C2CN(c3nnnn3C)C2)(C)C)CCN(C)CC1 58517,c1(C(=O)NCC(CNC(c2nc(CC)[nH]n2)=O)C)cc(C)ccc1[N+](=O)[O-] 58518,C1(C(N(C2CN(C(C3CCN(C)CC3)=O)CC2O)C)=O)CCc2nn[nH]c2C1 58519,c1(C(=O)NCCNC(c2c(C(N)=O)cccc2)=O)cnc2nccn2c1 58520,c1(C(=O)NC2CC(CNC(CCC3CC(C)C3)=O)CC2O)ccc(F)cc1C#N 58521,C1(N(C(=O)CN2C(=O)CNC2=O)C)CCCN(C(c2cc(=O)n(C)cn2)=O)CC1 58522,c1(C(N2CC(CNC(c3nc(CC)oc3)=O)C3C2C3)=O)cc(C)ccc1[N+](=O)[O-] 58523,c1(C(N2CCC(NC(C=CCN(C)CC)=O)C2)=O)cncc2c[nH]nc12 58524,N1(C(c2cocn2)=O)CCCCC1CCC1CCCN1C(C1CC=CC(O)C1)=O 58525,N1(c2c(OC)cnc(Cl)n2)CCC2(CC1)OCCC2NC(=O)C(C)OC 58526,C1(C(N(C2CC(NC(CCSC)=O)C2)C)=O)CCOCC1C 58527,c1(OC)c(F)c(C(=O)NCc2cccc(NC(C3CC3(C)C)=O)c2)cc(F)c1F 58528,N1(C(CC(C)(C)O)=O)CCN(C(=O)CCc2ccsc2)C(C(F)(F)F)C1 58529,c1(CC(N2C(CN(C(C(C)SC(F)(F)F)=O)C)CCC2)=O)ccccc1Cl 58530,n1(CC(N2CC(C)(CNC(c3c(OC)nn(C)c3)=O)C2)=O)cc(C)c(O)nc1=O 58531,c1(C(=O)NC2CC(CCNC(c3[nH]c(=N)sc3)=O)C2)n[nH]c2c1CC(F)(F)CC2 58532,c1(OC)cc(C(=O)NC2CC3(C2)CC(NC(=O)C(F)C2CCOC2)C3)ccc1C 58533,C1(CNC(C(Cc2c(C)nc[nH]2)O)=O)CCN(C(c2ncc(Br)cn2)=O)CC1 58534,C1(NC(CC=C)=O)CCC(CCNC(c2cn(C(C)C)nn2)=O)C1 58535,C1(C(=O)NCC(=O)NCC)CCC(O)CN1C(c1cn(CC)nc1C)=O 58536,N1(C(c2cn(CC)nc2)=O)CCCOC(CCNC(c2nccc(C)n2)=O)C1 58537,N(C(=NCCCNS(C)(=O)=O)NC1CCC12CCCCC2)CCN(C(C)=O)CC 58538,C1(CC=C)(NC(C2C=CCC2)=O)CCN(C(c2ccc(C(N)=O)cn2)=O)C1 58539,c1(C(=O)NCC2(C(F)(F)F)CCN(C(=O)OC(C)(C)C)C2)sc([N+](=O)[O-])cc1Cl 58540,N1(CC2CN(C(C=CC=CCC)=O)C2)CCN(C(c2cnsn2)=O)CC1 58541,C1(C(N2CCC(NC(CC(C)c3ccncc3)=O)C2)=O)COCCC1(F)F 58542,N1(C(c2cn(C)nc2Br)C(=O)N(CCC(=O)OCC)CC)CC=CCC(C)(C)C1 58543,c1(-n2ncc(C(=O)NCCCOCCCNC(C3C(C)C3)=O)c2)cccc(O)c1 58544,n1(CC)ncc(Cl)c1C(=O)NCC(C)CNC(=O)Cc1cc(C)[nH]n1 58545,C1(N(C(C=CSC)=O)CC(C)C)CCN(C(C2CCCCN2C(C)=O)=O)CC1 58546,C1(C(=O)NCC(CNC(c2cc(O)ccc2F)=O)O)CCC2(CCC2)O1 58547,C(C(F)(F)C(=O)NCCCCCNC(=O)CN1C(C)CCC1C)OC 58548,N1(C(CCC)=O)CCC(C)(C(=O)NCc2ccsc2)C1 58549,C1(C(N2CC(C(C)OC)C2)=O)CCC=CC1NC(C1CCCN(C)C1)=O 58550,n1(-c2c(C(=O)NCCN(C)C(C3(C)C=CCC3)=O)cccc2)ccc([N+](=O)[O-])n1 58551,c1(NC(NOCCC#C)=O)ccc(OCCc2ccccc2)cc1 58552,Cc1ccnc(C(=O)NCC2(NC(c3ccnc(CC4CC4)n3)=O)CCCC2)n1 58553,c1(C(C)NC(=O)CC2CSC2)nocc1C(=O)NCC1CCC(C)C1 58554,C=CCN(CC=C)N1CCC(CC(=O)N(CCCO)C)CC1 58555,CC(C)(C#Cc1cn(Cc2cscn2)nn1)NC(C1CCN2CCCC12)=O 58556,C#CCCC(O)C(=O)NC(C1CCN(C(C2CCS(=O)(=O)N2)=O)CC1)(C)C 58557,Cc1nc(NCCS(=O)C(C)(C)C)cc(NC(c2nccnc2C)C)n1 58558,C#CC1(O)CCN(C(C2CC(C)CN(C(C3(C#C)CC3)=O)C2)=O)CC1 58559,C1(C(CNC(C(C)OCC=C)=O)(C)C)CCCCN1C(=O)CN(CC)CC 58560,Cc1ncn2ccc(C(N3CC(CNC(=O)C=CC(C)C)C4(CC4)C3)=O)cc12 58561,c1(C(N2CC3(CC(CC(=O)NCCSCC)C3)C2)=O)cc(C)cc(Br)c1F 58562,CC(CC(=O)NC1(C)CCN(C(c2cccc3cnsc23)=O)C1)C(C)(C)C 58563,CCCN=C(NCC1(C)CCCc2ccccc21)N1CCC(OCC(C)C)C1 58564,n1(CCC)nc(C)cc1C(=O)NCC1CC(NC(C2(F)CC=CCC2)=O)C1 58565,C(CC(C)(C)C(=O)NCC1(F)CCN(C(C2(C)CCCC2(F)F)=O)CC1)OC 58566,c1(C(N2C(CNC(c3c(CC)nc(C)nc3)=O)CCC2)=O)ccc(C#N)c(O)c1 58567,C(=O)(CCC(C)(C)NC(=O)C1=COCCC1)NCCc1nc(C)sc1 58568,C(=O)(C(C)CN(C(=O)C(C1CCOCC1)O)C)NC(COC)CO 58569,C(=O)(C(C)CC(F)F)N(C(CC)CC(=O)NCCOC)CCOC 58570,c1(C(C)=O)cc(C(=O)NCC2CCN(C(=O)C(=Cc3cnn(C)c3)C)C2)oc1C 58571,c1(C(C(=O)NCC(O)CNC(C2(O)CCC2)=O)N(C)C)c(F)cccc1Cl 58572,C1(C(N(C2CCN(CC)CC2)C)=O)CC(C)CN(C(=O)CN2CC=CC2)C1 58573,N1(C(C(C)OCCCC)=O)CC2CCC2(CNC(=O)C=Cc2cnc(C)s2)C1 58574,c1(C(C(=O)NCC(CC)NC(=O)COCCN(C)C)O)cn(C)nc1C 58575,C1(COC)(NC(=O)C=Cc2ccnn2C)CCN(C(=O)CC(C)(C)OC)CC1 58576,c1(OC)nccc2c(C(=O)NCC3CC(CNC(=O)C4=CCCC4)CO3)c[nH]c12 58577,N1(C(CC=C=C)=O)CCC2(NC(=O)CCc3ccc(OCC)cc3)CCCC12 58578,C=CC1(CC(=O)NCCNC(c2ccoc2)=O)CN(C(=O)CC2CC3C=CC2C3)C1 58579,C=CCC(CC(C)C)C(=O)N(C1CCN(C(C2CC3(CC(OC)C3)C2)=O)C1)C 58580,C1(CNC(C2(C#N)CC(C)C2)=O)CCN(C(c2cnnc(Cl)c2)=O)C1(C)C 58581,C(=O)(C(F)(F)CCn1ccnn1)N1CC(OCCNC(c2ccnc(OC)n2)=O)C1 58582,C=CC1(c2nn[nH]n2)CCN(C(=O)C(N)Cc2cnc3c(c2)CCC3)CC1 58583,Cc1cc(OCC(=O)NCC(CO)NC(c2coc(C3CC3)n2)=O)cc(C)c1Cl 58584,C#Cc1ccc(OCC(=O)NCCN(CCC)C(c2conc2CC)=O)cc1 58585,Cc1cc(C(N2CCN(C3CC3)CC2C)C(=O)NCCC2(C)CC2)cnc1C 58586,C(=O)(C(C)CNC(c1cnc(O)o1)=O)N(CCC)C1CC1 58587,n1(CC)ncc(Cl)c1C(=O)NCC1CCCC1NC(C1(O)CC(C)(C)C1)=O 58588,c1(OC)cc(C(=O)NC2CCCCC2NC(=O)CCC2CC2C)cc(C)n1 58589,C1(NC(c2nccc(C)c2)=O)CC2CCC(C1)N2C(=O)CCCc1nc(C)cs1 58590,N1(C(=O)C(F)(F)F)CCc2nc[nH]c2C12CCN(C)C2.C1(C(=O)O)CCCCS1(=O)=O 58591,c1(C(=O)NC(CC)CN(C(=O)C(C)C2=CCCC2)C)oc2ccc(C)cc2c1C 58592,c1(C(=O)NCCN(CCCN(C)C)C(C2CC(O)C2)=O)n[nH]c2c1CCCC2 58593,CC1CCC=C1C(=O)N1CCCCC1CN(C(=O)C=Cc1cnc[nH]1)C 58594,CC1CN(C(C(=O)NCCN2CCOCC2)C(C)CC2CC(F)(F)C2)CC(=O)N1 58595,c1(N(C)C)ccc(C(=O)NCCC2(NC(=O)C(O)CN3CCCC3)CCC2)cc1 58596,C12(c3cn(CC(CC)C)nn3)COC(CN1C(c1nocc1Br)=O)C2 58597,c1(C(N(C2CN(C(=O)CCCN3C(=O)CNC3=O)C2)C)=O)n[nH]c2ccccc12 58598,N1(C(C(CCOC)NC(C(C)OCCOC)=O)=O)CCCC(O)(C2CC2)C1 58599,c1(C(=O)NC2C(C)(C)C(CNC(=O)CN3CC4CC4C3)C2)cc2sccc2s1 58600,C1(C(=O)NC2(CO)CC(F)(F)C2)(CC)CCCN1C(=O)Cc1ccsc1 58601,Cc1ccc(Cl)c(O)c1C(=O)NC1CCN(C(=O)CC(F)(F)F)CC1C 58602,C(C)(CNC(C1CC(=O)N(c2nccs2)C1)=O)(C(C)C)NC(CSC)=O 58603,C(=O)(C(C(C)(C)C)NC(=O)OC)N1CCC(F)(CNC(c2cn(CC)nc2)=O)C1 58604,CC1(C)OCC2CC12NC(C1(NC(c2cc(Cl)n[nH]2)=O)CC(F)(F)C1)=O 58605,C1(COC)(CNC(CCOCCCNC(=O)CNC(=O)OC(C)(C)C)=O)CCCC1 58606,CC(C)(CCNC(C1CCC(F)C1)=O)NC(=O)COCCN(C)C 58607,c1(C(=O)OC)ccc(CNC2CC2C(=O)NC(C)CC#N)c(Br)c1 58608,c1(NC(N2C(CC(=O)NC(CSCC(=O)OCC)=O)CC2)=O)ccc(NC)cc1 58609,Cc1ccc(O)c(C)c1NC(=O)C(CCNC(N)=O)NC(C1CCC(C2CC2)C1)=O 58610,c1(C(=O)NCCN(C(=O)CC2CN(C)CC2O)CC)ccc2c(c1)OC(C)(C)C2 58611,N1(Cc2c(C(=O)OC)c(C)sc2)CC2CS(=O)(=O)CC2(C#N)C1 58612,CNS(=O)(=O)NCC(=O)NCCN(C(=O)CCn1ncn(C)c1=O)C1CC1 58613,C12(C(N3CCN(C(c4c(C)coc4)=O)CC3CO)=O)CCC(N(C)C)(CC1)CC2 58614,C1(C(C#C)C)CCN(C(C23CC2CCN3C(=O)C(O)C2CC2)=O)CC1 58615,N1(C(CCCC(C)C)=O)CC(NC(=O)CCC2(C)CC2)C2CCCC12 58616,C(=O)(C(C)(C(F)(F)F)Oc1ccccc1)N1CCCN(C(C(CC)(C)O)=O)CC1 58617,CC1(C)C2CCC1(CC(N1CC(CNC(C3SCCCS3)=O)C1)=O)CC2 58618,CC(C(=O)N(C)CC1CCN(C(C2CCCC2)=O)C1)C(C)(F)F 58619,CCCC(C(=O)OCC)N1CCN(C(=O)C(C2CCCCC2)N)CC1 58620,C1(NC(C2N(CC)CC2)=O)CC2CCC1(NC(c1cnn(CC)c1Cl)=O)C2 58621,c1(C(=O)NC(CCNC(C2N(CC)CCOC2)=O)C)ncc(Br)cc1F 58622,c1(C(=O)Nc2cncc(Cl)n2)ccc(=O)n2c1COCC2 58623,C1(C)(CNC(C(CN(C)C)O)=O)CN(C(=O)C(C)(C)NS(C)(=O)=O)CCO1 58624,C=C(Cl)CC(C(=O)N1CC(CO)C2(CC2)C1)NC(c1cc[nH]c1)=O 58625,N1(C(CC(C)F)=O)CCN(C(c2cc(Br)cn3ccnc23)=O)CC2(CC2)C1 58626,C(=O)(C1=CCN(C(c2cn(C)c(=O)cn2)=O)C1)NCC1(C(=O)OCC)CC1 58627,N1(C(c2ccc(-c3ccc(S)cc3)cc2)=O)CCCC2CNCCCC12 58628,c1(C(C(=O)NCCN(C(=O)CCc2cnoc2)CC(C)O)O)ccc(Cl)cc1 58629,C1(CNC(C2(CC)CC2)=O)(COC)CCCN1C(C1CC(SC)CN1C(C)=O)=O 58630,N1(C(Cc2cnc(C)[nH]2)=O)CC2OCCN(C(=O)CC3C=CCC3)C2C1 58631,c1(CC)nn(C2CC2)cc1C(=O)NCCNC(c1cncnc1)=O 58632,c1(OCC)ccc(C(=O)NC(CNC(c2cscc2CC)=O)CO)cc1C 58633,Cc1nc2ccccc2cc1C(=O)N(C1CCCC(N(C)C(C2COC2)=O)C1)C 58634,N1(C(C2(CS(C)(=O)=O)CCC2)=O)CC2CCC2(NC(C2COCCC2(F)F)=O)C1 58635,C=C(C)CCCC(=O)NCC(C)N(C)C(c1ccn(C(C)C)n1)=O 58636,Cc1ccc(C(=O)NCCC2(O)CCCN(C(c3nnc(S)n3C)=O)C2)c(N)n1 58637,N1(C(C(CCC)CCC)=O)CC(CO)C2(C1)CN(C(=O)C(CC)n1ccnc1)C2 58638,C1(C(N2CCC(COC)(CNC(c3cnc(O)s3)=O)C2)=O)CCC(C)=C(C)C1 58639,C1(c2n(C(CC)(C)C)nnn2)(Nc2ccc3c(c2)OCO3)CCCC(C2CC2)C1 58640,c1(C(=O)NC2CC3(C(NC(C4CC(CCC)C4)=O)C3)C2)ccc2c(c1)C(=O)CCC2 58641,CCC(CCC(=O)N1CCC(n2cccn2)C1)NC(c1cnnc(O)c1)=O 58642,N1(C(C=CCCC(C)C)=O)C(C(=O)NC2(C)CCCOC2)CCC12CC2 58643,C1(NC(C2(C(=O)NC)CC2)=O)CCCN(C(c2ccnc(C(C)C)n2)=O)C1C 58644,C=CC1CN(C(C2CC(C(F)F)(OC)C2)=O)CC1NC(C1CCCCCCC1)=O 58645,CC1(C)C=C(C(=O)NC2CCC(NC(C3(F)CCCCCC3)=O)CC2)C1 58646,C1(C(=O)NC(CC)C(O)c2ccccc2)CCc2cnn(CCCC)c2C1 58647,C(C)(c1ccc2ccnnc2c1Cl)=CCCC 58648,C1(CNC(c2cn(CC=C)nn2)=O)CN(C(=O)C=CC(=O)NC2CC2)CCC1C 58649,C#CC1(C)CCCN1C(=O)Cc1cc(=N)[nH][nH]1 58650,N1(C(C2(CCCC)CC2)=O)CCC2C(CCN2C(C2C=CCS2)=O)C1 58651,C1(C(=O)NC2CCN(C(c3nocc3C3CC3)=O)C2)C2CCCOC12 58652,C=C(Br)CC(C)(C)C(=O)NCCC1CCC(NC(C2(OC)CC2)=O)C1 58653,C12(NC(C(c3ccccc3)C)=O)CC(C1)N(C(=O)C(C)N1CCCC1)C2 58654,C(=O)(C1Cc2ccc(F)cc21)NCC1CC(N)(C(C)C)C1 58655,C=CC(C)(CCOC)C(=O)NC(CN(C)C)C(=O)NCC(C)(C)CN=[N+]=[N-] 58656,N1(C(c2c(F)ccc(OC)n2)=O)CCCCCC(NC(c2cncc(F)c2)=O)C1 58657,c1(C(=O)Nc2ccc(C(=O)NCc3n(C)ccc3)cn2)c(F)cc(O)cc1F 58658,c1(NC(C(=O)NCC(C(C)O)C)=O)nc2c(s1)C(=O)NCC(C)(C)C2 58659,Cc1nccn1CCCNC(c1nnnn1C1(C)CC1)C1CCCCC1 58660,CC(C)CC(CNC(c1cc(CO)[nH]n1)=O)C(=O)NC1CC(CO)C1 58661,c1(C(=O)NCC(c2ccccc2)CNC(CC=C)=O)ccc2c(c1)C(=O)NC2=O 58662,N1(C(C(C)CO)=O)CCCC2(NC(C3(CN(C)C)CC3)=O)CC2C1 58663,FCCCN=C(NCC1(c2ccc(Cl)cc2)CC1)NCC1CC=CCO1 58664,C(=O)(C(C)C(C)NC(=O)CC1CN(C(=O)C(c2cncn2C)O)CC1C)OC 58665,C1(C(=O)NCC(=C)C(F)(F)F)CC(NC(=O)CCC#CC)C12CCC2 58666,c1(C(N(CC(CNC(c2c(C)coc2C2CC2)=O)C)C)=O)ccc2c(c1)CCN2 58667,c1(C(=O)NCCC(=O)N2CC(OCC(=O)NC3CC3)C2)ncncc1Cl 58668,Cc1oc(CNC(C2CCCC(F)C2)=O)nc1C(=O)NC(c1ccc(O)cc1)C 58669,CC1(NC(=O)CC2CCCC2(F)F)CCCN(C(c2cnc3c[nH]nc3c2)=O)C1 58670,Cc1nc(N(C)CC2CCCN(C(c3ccco3)=O)C2)cc2nncn12 58671,C1(CC(=O)N(CC=C)CCO)(OC)CN(C(=O)CCc2nc(C)no2)C1 58672,c1(CC(=O)N(C(CN(C(C=C(C)Cl)=O)C)C)C)cccc(OCC#N)c1 58673,C(=O)(CCCS(C)(=O)=O)NCCOC(C)(C)CNC(c1cc(C2CCC2)no1)=O 58674,N1(C(C(C)SCCCC)=O)CC2C(C(N3CCC(c4ncco4)C3)=O)C2C1 58675,C12(NC(C3C(CNC(CNC(C)=O)=O)C3)=O)CC1COC2(C)C 58676,c1(C(=O)NC2C(C(=O)NC(CCCCC)C)OCC2)cc(C#N)n(C)n1 58677,NS(=O)(=O)c1cncc(C(=O)NC2CCCN(C(=O)C=C3CCCC3)C2)c1 58678,CC(CCCNC(=O)CNC(=O)C(C)(C)F)NC(=O)NCc1ccccc1 58679,C1(C(=O)NCC=C)CCC(NCc2csnn2)CO1 58680,c1(C(N2CCOCC(CNC(C3(C)CCCCC3)=O)C2)=O)ccc(Cl)c(N)c1Cl 58681,N1(C(C(C)O)=O)CCCC(CNC(=O)CC2COC(C)(C)C2)C1 58682,c1(C(=O)NC(CNC(CS(=O)(=O)NCC)=O)(C)CO)ccn2nccc2n1 58683,Cn1ncc2cc(C(=O)NC3CCCOC3CN)cc(O)c12 58684,c1(C(N2CC(O)CC(NC(CCSCCC)=O)C2)=O)c(F)ccc(OC)c1OC 58685,N1(C(c2ncn(CC)c2)=O)CCCN(C(C2(C)CC2(C)C)=O)CC1C(C)C 58686,C12(NC(=O)C3=COCCC3)CCCCCC1N(C(C1C=CCC1)=O)CC2 58687,c1(C(=O)NCC2CCC(CNC(C3CC3CF)=O)CC2)c(O)cccc1Cl 58688,N1(C(c2c(C)cccc2)=O)CCN(C(C2(C(F)F)CCCO2)=O)CC1C(F)F 58689,C1(F)(CNC(C(C)SC(C)C)=O)CCCN(C(C2CC(O)C2)=O)CC1 58690,Nc1cnccc1C(=O)NC1CCC(NC(c2ccnn2C2CC2(F)F)=O)CC1 58691,c1(OC)ccc(CCCCNC(=O)NC2CCC(c3nc(C)no3)CC2)cc1 58692,CC(C)CCCCC(=O)N1CCC(C2CCCN2C(c2cc(Br)n[nH]2)=O)C1 58693,C1(C)(NC(Cc2cc(C)sc2C)=O)CCCN(C(C2CCCCC2(F)F)=O)C1 58694,c1(C(N2C3CC(CNC(CSCCOC)=O)C(C3)C2)=O)cc2ccccn2c1 58695,c1(C(N2CCC(C(CO)NC(CCSC)=O)CC2)=O)cn2ccnc2s1 58696,Cn1nc(C(N2CCCC2CNC(=O)CC2C=CCCC2)=O)cc1F 58697,C(=O)(CC(C)(C)C(F)F)N1CC2(COC)CC1(CNC(=O)C#CC(C)C)C2 58698,C1(NC(C2C3(CC3)C23CC3)=O)CC2CC(NC(C3CCSCC3)=O)C1C2 58699,c1(C(=O)NCC(CNC(c2c(C)cco2)=O)(C)O)noc2ncccc12 58700,N1(C(c2nc(C(F)(F)F)n[nH]2)C(=O)NCCOC)CC2C(=O)N(C)C(=O)C2C1 58701,Cc1[nH]nc(C(F)(F)F)c1C(=O)NCC1CN(C(=O)CC2CC2C2CC2)CCO1 58702,c1(CC(=O)NCC2(C)C(C)CN(C(C3COCCO3)=O)C2)cccc2c1CCC2 58703,c1(CNC(c2csc(-c3ccccc3Oc3ccccc3)n2)=O)ccnc(F)c1 58704,C12(C(=O)NC(C(=O)NCC=CC)c3ccco3)CCCN(CC1)C2 58705,C1(NC(C(CCO)N(C)C)=O)CCN(C(C2CCCS2)=O)CC1O 58706,N1(C(Cc2c(CC)cccc2)=O)CC2CC1CCC2NC(c1cnsc1)=O 58707,C1(NC(C(F)=CCC)=O)(COC)CCN(C(=O)C(C)Cc2cnc[nH]2)C1 58708,C(C1CCCCC1)=CC(=O)NC1C(NC(CCc2cc(C)[nH]n2)=O)CC1 58709,c1ccc(Cl)cc1.c1(NCC(COCC)O)noc(CN(C)C)n1 58710,N(C(=NCCC(C)(C)C#N)NCC1CCCC(CC)C1)CC(C=C)(C)C 58711,c1(C(=O)NC(C2CCCN2C(c2cc(F)ccc2N)=O)C)ccc(S(C)(=O)=O)o1 58712,C1(N(C(C=CCN(C)CC)=O)C)CCN(C(c2c(C(F)(F)F)coc2C)=O)CC1 58713,CCCCC(F)C(=O)N1CC(OCCC(=O)Nc2cccc(COC)n2)C1 58714,S(=O)(=O)(c1ccc(NC2CCOC3(CCCC3)C2)c(F)c1)NCC(C)CO 58715,CC1CC2(CC(C(=O)NCC3(C)CCCN(C(c4ccc(=N)[nH]c4)=O)C3)C2)C1 58716,C1(NC(c2cc(C)sc2C)=O)CCC12CCN(C(c1ccc(O)cc1)=O)CC2 58717,C1(NC(C(C)NC(C(=Cc2ccco2)C)=O)=O)COC2(CCC2)C1 58718,CC1(C)CCCC(O)(C(N2CCC2CNC(=O)CC2CC2(C)C)=O)CC1 58719,CC1(C)C(CC(=O)NCCNC(=O)CNC(c2ccco2)=O)CC1O 58720,CC1(C)COC(C(=O)NC2CCCC(CNC(c3cc(Cl)ccc3Cl)=O)C2)CO1 58721,C1(C(=O)NC(C2CN(C(c3cccc(O)n3)=O)C2)C)C2CCC1(c1ccco1)C2 58722,C1(C(N2CCCC(CO)C2)=O)CCCC12CCN(Cc1cc(F)c(Br)cc1F)C2 58723,Cc1[nH]c(C#N)cc1C(=O)NCC(C)(C)NC(=O)Cc1ccc(F)cc1 58724,C(CCNC(=O)CCc1cc(C)no1)(C(C)C)NC(COC(CC)(C)C)=O 58725,C(=O)(CC(CNC(c1cc(C2CCCN2)no1)=O)OCC)N(CC(C)C)CCC 58726,C(=O)(C(C)CC(F)(F)F)NCCCN(CCCNC(=O)C(c1ccnn1C)O)C 58727,C(C(C(C)(C)C)NC(c1cc(C)n(C2CC2)n1)=O)NC(CCSCCC)=O 58728,C(=O)(CCCC(=O)N1CC(N(C)C(C2CCC(C)O2)=O)C(O)C1)N(CC)CC 58729,CN1CC(C)(C)CC1C(=O)NC1CCCC1CNC(c1cc(Cl)cs1)=O 58730,c1(OC)cc(OCC(N)=O)ccc1NC(C1CC(C(=O)O)C1N)=O 58731,N1(C(C2CC(SC)C2)=O)CCC(NC(C2CN3CCC2CC3)=O)C(O)C1 58732,N1(C(c2c(C#C)cnn2C)=O)CCC2(CCCN2C(C23CCCC2CCC3)=O)C1 58733,C1(O)(C(=O)NCC2N(C(c3cnc(Cl)s3)=O)CC(C)(C)OC2)CN2CCC1CC2 58734,c1(NC(C(C)N(C)C(=O)OC(C)(C)C)=O)c(O)nn(C)c1C(F)(F)F 58735,c1(OC)cc(CC2CC2C(=O)Nc2nc(C)c(C)s2)cc(I)c1OC 58736,C1(CC(=O)NC2CCC(NC(CC3CN(C)C3)=O)C2)CCC(C(F)(F)F)CC1 58737,c1(C(c2n(C(CC)C)nnn2)NCCc2nccs2)cc(Cl)ccn1 58738,C1(C(=O)NC2(CCNC(C3(CC(C)C)CC3)=O)CC2)CC(=O)N(C2CN(C)C2)C1 58739,CCCC(C#N)C(=O)NC(C(=O)NOC(C)(C)C(=O)OC)C1(C)CC1 58740,c1(N2CCCC(OCC=C)C2)nc(=N)[nH]c(=NCCc2ccc(CSC)cc2)[nH]1 58741,CC1CC=C(C(=O)N2CCC(F)CC2C(=O)NOCCF)CC1 58742,C(=O)(C(CC(C)C)C(C)C)NC(CC)(CNC(c1nnn2c1CSCC2)=O)CC 58743,C1(NC(c2c(CC)n(C)nn2)=O)CN(C(c2cnn(C)c2F)=O)CC12CC2 58744,C#Cc1ccc(C(=O)NC2CC3CCC(C2)N3C(=O)CC2CCOC2)cc1F 58745,C1(F)(C(=O)NCCN(C)C(c2cncc(-n3cncn3)n2)=O)CCOCC1 58746,Cc1ccc(C(=O)N(CCC(=O)NC(C)CCC2CCCO2)C(C)C)c(O)c1 58747,N1(C(c2c(CC)cns2)=O)CC2(C(=O)O)CC1CCO2 58748,C1(CNC(C2(CCOC)CCC2)=O)C(C)CCN1C(C1CC1C)=O 58749,C1(C(=O)OC)CN(C(=O)NCCCN2CC3CC3C2)C2(CCC2)C1 58750,Cc1cccc2c1CC(C(=O)NC1COCCN(C(=O)C(F)=C3CCCC3)C1)O2 58751,N1(CC)CCCC1CC(=O)NCC(C)(C)CNC(=O)C=CC(C)CC 58752,C(=O)(CCC(=O)N1CC(c2ocnc2C(=O)NCC2COCCO2)C1)NC 58753,c1(OC)coc(C(=O)NCC2(C)CCCN2C(=O)COCCN(C)C)cc1=O 58754,C1(OCC)CCCCC1NC(=O)C(O)CCNC(=O)CCc1nccs1 58755,C1(NC(C23C(CN(C(=O)C=Cc4cc[nH]c4)C2)C3)=O)CC2(CCCO2)C1 58756,C1(O)(CCNC(c2c(C)nsc2)=O)CCN(C(=O)C(C)Cc2cnc[nH]2)CC1 58757,C(=O)(CCCC(=O)NC1CN(c2ncc(Cl)c(O)n2)CC1(C)C)NCC 58758,c1(OC)ccc(C(=O)NC2CCN(C(C3CC3(F)F)=O)C2C2CC2)c(O)c1 58759,C1(C(=O)NCCN(C(CNC(c2cccc(C)c2)=O)=O)C)CCC2(CCOC2)O1 58760,C1(C(N(C(C)CCNC(c2ccc(-c3ccco3)[nH]2)=O)C)=O)CC2(C1)CC21CC1 58761,N1(C(C(CSC)C)=O)CCN(C(C2CCC(=O)N2C(C)C)=O)CC1c1cn[nH]c1 58762,C12(CNC(=O)NCCCC3CCCCO3)CCC(CO1)C2 58763,c1(C(=O)NCC2(CNC(C(C(C)C)OCC)=O)CCOCC2)cn(C)c(=O)n1C 58764,c1(C(N2CCC(O)(CNC(COCCOCC)=O)C2)=O)ccc(C2CC2)cc1F 58765,C1(C(=O)OC)CC(Oc2ccc3cc2-3)C12CCOCC2.C(C)(C)(C)OC 58766,C1(c2ccccc2)(CNC2C(F)(Br)C2)CCCC1 58767,N1(C(C2C(CC)C2)=O)CC2CCN(C(C3C(C=C(C)C)C3(C)C)=O)CCC2C1 58768,C1(CN2CCC(NC(COC(CC)C)=O)C2)CCOC(C)C1 58769,c1(NCC(=O)N(CCN(C(C)C)C(C2CC(C)OC2C)=O)C)ccc(N)cc1 58770,c1(SCC)nccnc1C(=O)NCC1(CSC2CC(CC(C)(C)C)C2)CCCO1 58771,c1(OC)ccc(SCCC(N2CC3CC3(NC(C34CCC(C3)C4)=O)C2)=O)cc1 58772,CC1(CNC(C2CC2C)=O)CCN(Cc2cccnc2Cl)CC1 58773,C#Cc1ccccc1CC(=O)NCC1C2CC1N(C(=O)C(C)(Cl)Cl)C2 58774,c1(N(c2ccccc2F)CCNC(C(CC)N(C)C)=O)nc(C2CC2)nc(=N)[nH]1 58775,c1(N2CC(c3ccc4occ(C)c4c3)OCC2)ccn2ncc(S(=O)(=O)NC)c2n1 58776,N1(C(C(CCC)CN)=O)CCC2CCCCC2CC1 58777,C1(=CC(=O)NC2CCN(C(c3ccc(F)s3)=O)C2)CN2CCC1CC2 58778,C12(CNC(c3ccn(CCNC(C(CCC)F)=O)c3)=O)CCCN(CC1)C2 58779,Cc1nn(CC(=O)NC2CCN(C(=O)CSC(C)(C)C)C2C)c(C)c1Cl 58780,CC1CC(NC(=O)C(=O)NCC2CC2)CN1C(c1cnc(C(F)F)nc1)=O 58781,CC(C)C(C(F)(F)F)NC(C1CC=CCN1C(c1ccc(Cl)s1)=O)=O 58782,N1(C(c2ncn(-c3ccn(C)n3)c2)=O)CC2CCN(C(c3csc(=N)[nH]3)=O)CC12 58783,C=CC(C)C(C)C(=O)NCC1(CNC(c2cn(C)c(-c3ccccn3)n2)=O)CC1 58784,N1(C2CCCN(C(CSCC=C)=O)C2)CCN(C(C2CC(N(C)C)C2)=O)CC1=O 58785,N1(C(C(Cc2ccoc2)NC(c2ncc(F)cc2F)=O)=O)CC2CC1CC2O 58786,C1(F)(CNC(Cc2ccc(C)s2)=O)CCN(C(=O)CCC2CCCCO2)C1 58787,N(C1CCCc2cc(F)ccc21)C(N1C(CCC)(CO)CCC1)=O 58788,C1(N(C(c2c(C)non2)=O)CCO)CCCN(C(=O)C(F)CC2CCCCC2)C1 58789,c1(C(=O)NCC2CC(NC(C(C(CC)C)C)=O)C2)c(C)ccc2ncccc12 58790,Cc1nnc(CCCC(=O)N(CC(O)CNC(c2ccc(CO)cn2)=O)C)n1C 58791,Cc1nc(CC(=O)NC(CC2CC2)C(=O)NC2CC(CC(C)(C)C)C2)n[nH]1 58792,C(=O)(CC(C)C(=O)NCc1cc[nH]c1C(=O)NCc1ncnn1C1CC1)OCC 58793,CN1CCC(n2cc(CNC(C3CC3)=O)cn2)CC1.C1(CNC=O)(CF)CCC1 58794,N1(C(C2CNC(=O)N2)=O)CC(NC(c2csc3cncn23)=O)C2CCCCC12 58795,C(=O)(CC(C)(C)C(C)(F)F)NCCNC(C1N(C(C)C)CCC1)=O 58796,c1(C(N2CCC(OCCNC(c3c(C)c[nH]n3)=O)C2)=O)ccc2ncnn2c1 58797,c1(CCN(C)C(=O)OC(C)(C)C)cnn(C)c1.c12cnc(s1)NCC2 58798,N1(C(Cc2nc(C)sc2C)=O)CC(N(C)C(C2C=CCC2)=O)C2(CC2)C1 58799,C1(C(C)NC(C2CNC(=O)O2)=O)CCCCN1C(c1c[nH]nc1OCCOC)=O 58800,C(=O)(C#CC1CCC1)NC(C(=O)NCC(CC)C(C)C)COC 58801,C1(CCN(C(Cc2cc(C)[nH]n2)=O)CC2CC2)CCN(c2nnc(CO)s2)CC1 58802,c1(C(=O)NCC(CNC(C2C(CC)C2)=O)O)ccc2nn[nH]c2c1 58803,CC(CC(C)NC(=O)Cc1csc(C(F)(F)F)n1)NC(=O)C(F)(F)C1CCCC1 58804,N1(C(c2ccc(C=C)cc2)C(=O)NCCC)c2ccccc2C(C)C1C 58805,C(CNC(=O)Cc1ccc(F)cc1F)(CC(F)(F)F)NC(c1c(C)[nH][nH]c1=N)=O 58806,C1(CNC(CSCC)=O)CCCCCN1C(c1oc(CC2CC2)nc1C)=O 58807,N1(C(C(CCN(C)C)O)=O)CC2CC(NC(=O)CCc3cnccn3)CC1C2 58808,c1(N2CCC(N(C(C3C(=C)C3)=O)C)C2)nc(C(C)C)ccc1C#N 58809,C1(C(=O)NCCOC2CCCC2)CCC2CCC1N2C(=O)Cc1ccccn1 58810,C1(C(C)NC(=O)C=CC2CCC2)CN(C(C2(C(F)F)CC2)=O)CCO1 58811,c1(C(=O)NCCOCCNC(=O)CC(n2cnnn2)C2CC2)ccc(Cl)cc1 58812,c1(NC(C2(CNC(C=Cc3ccc(C)s3)=O)CC2)=O)ccc(C)c(Cl)c1 58813,C(=O)(C(CNC1CC1)Cc1ccc(Cl)cc1)OC.c12ncc(s1)c(=O)[nH]2 58814,N1(C(C2(COC)CCCC2)=O)CCC(CNC(C2C=CCCC2)=O)(OC)C1 58815,c1(NS(C)(=O)=O)cc(NC(=O)NCCCn2cnnc2)ccc1F 58816,N1(C(C2N(CC)CCC2)=O)CCC(CC(=O)NC2CCC(=O)N(C)C2)C1(C)C 58817,CN1CC(C(=O)N(C)CC2CCN(C(c3cnn(CC(F)(F)F)c3)=O)C2)CC1=O 58818,N1(C(=O)NC(C)(C)C)CCOC(C(=O)N(CC#N)Cc2ccc(Cl)cc2)C1.N1CCCC1 58819,CSC1=C(C(=O)NC2CCC(CCNC(=O)CCN3CCOCC3)C2)CCCC1 58820,Cc1occc1C(=O)NCC(C)C(=O)NCC(=O)NC(C)C 58821,C1(C(=O)NCCc2n[nH]cc2C(=O)NC(C)C(C)SC2CC2)(CC)CCOC1 58822,C(=O)(C(C(C)NC(=O)CCc1ncnn1C)C(C)C)NCc1nccc(C)c1F 58823,N1(C(C2CC=C(C)CC2)=O)CC2(CCC2NC(c2cc(Cl)no2)=O)C1 58824,Cc1cccc(O)c1C(N1CC(N(C(=O)C(C2CCOCC2)C)C)C(C)(C)C1)=O 58825,S(=O)(=O)(c1ccc(NCCc2cc(C(F)(F)F)co2)c(Cl)c1)NC1CC(C)C1 58826,C(CC(=O)N(C)CCNC(=O)C(C)C)N(C(=O)C(C1(C)CC1)N(C)C)CC=C 58827,C1(O)(CNC(c2n(C(C)C)ncc2)=O)CCN(C(=O)CN2C(=O)CCC2=O)C1 58828,N1(C(C(C(C)C)SC)=O)CCC(C2CCN(C(=O)COC(C)C)C2)CC1 58829,C1(C(=O)O)C2CC1N(C(=O)CN1CCCC1)C2.O=C(C(F)CC1CCOC1)N1CCCC1 58830,CC(CN(C)C)C(=O)NC1CCC(CNC(C2(C)CC2Br)=O)C1 58831,C1(C(=O)NCC(CCNC(c2cnc(C3CC3)[nH]2)=O)OC)C(C#N)C1(C)C 58832,Cc1c(N(CCCN2CCN(C)CC2)C)ncnc1N1CCCC2(CC2)C1 58833,c1(NC(N2CCCC(NCCc3sccc3F)C2)=O)cccc(C(F)(F)F)c1F 58834,c1(C(N(C)CC2CN(C(=O)C(C)(C)C3CC3)CCO2)=O)ccc2scnc2c1 58835,C1(NC(C(C)OCCOC)=O)(COC)CCN(C(c2cnc(C)s2)=O)CC1 58836,N1(C(C(C)OC)=O)CCCCC2(CCN(C(c3cnn4ccncc34)=O)C2)C1 58837,c1(C(C(=O)N(CC(C)O)CCNC(C2(OC)CC2)=O)OC)ccccc1 58838,Cc1ncccc1C=CC(=O)NCCC1CN(C(=O)COC2CCC2)CC(C)O1 58839,C1(COCC#C)CCN(C(C2(CC)C=CCC2)=O)CC1 58840,C(=O)(C(F)n1ccnc1)NCCCN(C(C1CCSC1)=O)CC 58841,C#CCC(C)(CC)C(=O)NCCC1CCN(C(=O)Cn2[nH]cnc2=N)CC1 58842,CCC(CC(=O)N1CC(F)(CNC(C23CC2COC32CCC2)=O)C1)CC(C)C 58843,c1(C(=O)NCC(C)N(C(=O)CC(C(F)F)n2ccnc2)C)cc(O)ccc1OC 58844,Cc1cnc(F)c(CNC(C23CC(NC(=O)C(F)(F)CN(C)C)(C2)C3)=O)c1 58845,C1(NC(C(COCc2ccccc2)OC)=O)(CO)CCN(C(=O)COC)C1 58846,C#CCC(C)(C)C(=O)NCC1CCC(C(N2CCCCCCC2)=O)C1 58847,C1(OCC)CC2(C1)CC2C(=O)N(C)CCNC(=O)CCc1ncc(C(C)(C)C)o1 58848,Cc1c(F)ccc([N+](=O)[O-])c1NC(C12CC1CN(C(c1ccccc1I)=O)C2)=O 58849,Cc1csc(CCCC(=O)NCCC2CC(NC(C3(C)CCOC3)=O)C2)n1 58850,C1(C(N2CC(NC(Cn3ncc(C#C)c3)=O)CC(C)C2)=O)(OC)CCC(C)(C)C1 58851,C1(C(=O)NC2(C)C(C)CCC2)CCOCCN1C(=O)C(O)CN1CCCC1 58852,N1(C(CSCCC)=O)CCC(CN(C)C(C2CC(O)(CCC(C)(C)C)C2)=O)C1 58853,c1(-n2cc(C3CN(C(C(C=C)(C)O)=O)C3)nn2)cccc(C)c1Br 58854,N1(C(N(C)CCC2CC2)=O)CCC(C(=O)O)C(c2cnn(C)c2)C1 58855,C(=O)(C1=CCCOC1)N1CCC(COC)(NC(=O)CC2CCCN2C)C1 58856,c1(-c2ccn(CC)n2)cnc(NC(c2ccsc2C(F)F)=O)c(O)c1 58857,C(CNC(c1nc(C(F)(F)F)oc1C)=O)(CC(F)(F)F)NC(C(C#C)(C)C)=O 58858,CCC(C)C(O)C(=O)NC1(CF)CCN(C(=O)CCN(CCCCOC)C)C1 58859,c1(C(N2CC(C(=O)Nc3ccnc(C)n3)OCC2)=O)cc(F)c(F)cc1F 58860,C12(CCNC(CCCC#N)=O)CCC1CN(C(c1cnc(O)o1)=O)C2 58861,c1(NC(=O)C=CC(=O)OCC)ccc(C(N2CCC(CCC=C)C2)=O)cn1 58862,c1(COCC)nc(N2CCCC2CN(C)C(c2cnc(C)s2)=O)cc(C)n1 58863,c1(C(=O)NC2C(NC(c3cc(C)sc3)=O)CCCC2)cc(F)cc(F)c1F 58864,c1(NCC2C(C)CCN(C(C3CCCSC3)=O)C2)cccc(F)c1[N+](=O)[O-] 58865,CC(N=c1[nH]c(N2CCOC(C3CCCC3)C2)nc2c1SCC2)c1ccncc1 58866,C1(NC(c2c(C)cno2)=O)CN(C(=O)C(C)(O)CC(C)C)CC12CCOCC2 58867,C1(OCCC)CCCN(C(C2(C(C)NC(c3cnc(C)o3)=O)CC2)=O)C1 58868,c1(C(c2nnnn2CC)NCC(=C)F)ccc2ccccc2c1Br 58869,CC(CC1=CCCCC1)(c1nnnn1C)NCc1cc(F)c(C2CC2)c(F)c1 58870,CC1(C)CN(C(=O)NC2CCCC3CC23)Cc2cccc(OC)c2O1 58871,C1(C(=O)NC(CNC(=O)OC)C)CCC2CCC1N2C(c1cnc(Cl)n1C)=O 58872,C1(CNC(C=CC=CC)=O)CN(C(=O)CCc2ncccn2)C(C)(C)C1 58873,C1(CNC(C(COC)O)=O)CCCC12CCN(C(c1cn(C)ccc1=O)=O)CC2 58874,C1(CCc2n(CC=C)nc(-c3ccccc3Cl)n2)CC(OCC)C12CCC2 58875,c1(-n2cc(C3N(C(C(C)OCC(C)C)=O)CCC3)nn2)c(F)cccc1Cl 58876,Cc1nc[nH]c1CC(=O)NCCOCCN(C(=O)CC1CS(=O)(=O)C1)C 58877,c1(C(=O)NC(CC)CNC(=O)Cc2cn(C)nn2)c(C)noc1C 58878,C1(C)(C(=O)NC(CNC(CC2N(C)CCCC2)=O)C2CC2)CCC2CC2C1 58879,N1(CCN(c2ccc(C(F)(F)F)cc2)C)C(=O)CCN(CCCCCCO)C1=O 58880,C1(NC(c2cn(CCN(C)C)nn2)=O)CC(CNC(C2C=CCCC2)=O)C(O)C1 58881,c1(C(N2C(CNC(c3ccc(OC)nc3)=O)C=CC2)=O)cnn2c1OCCC2 58882,C(CNC(c1nc(C)oc1C)=O)(C(C)C(C)C)NC(CCCC)=O 58883,C1(CNC(C=C(CC)C)=O)CC2CCC(C1)N2C(=O)Cc1csc(Br)c1 58884,C1(CNCCc2c(C)c(Cl)ccc2)CCC2(CCCOC2)O1 58885,C1(O)(CN(C(C(C)c2cc[nH]n2)=O)C)CCN(C(=O)CCn2ncn(C)c2=O)C1 58886,N1(C(CC=CC=C)=O)CCCC2CN(C(c3cc(Br)ccn3)=O)CCCC12 58887,Cc1ccnc(C)c1C(=O)NC1CCCCC1NC(C1(C(F)F)CCCO1)=O 58888,N1(Cc2cc(OC)c(Br)cc2)CCC(F)(F)C(C(=O)N=c2cc(C)o[nH]2)C1 58889,CC(C(=O)NC1CN(C(c2ccc([N+](=O)[O-])c(O)c2)=O)CC1O)C(F)(F)C(F)F 58890,Cc1cn2cccc(C(=O)N(C)CC3(NC(c4cnoc4C4CC4)=O)CC3)c2n1 58891,c1(C(c2n(C(CC)(C)C)nnn2)NC2C=CCCC2)ccc2scnc2c1 58892,C1(CC(N2C(C)(CCC)CC2)=O)CN(C(c2cc(F)ccc2O)=O)CC12CC2 58893,CC(CC(C)(F)F)C(=O)NC1COCC1NC(c1cccc2c1COC2)=O 58894,C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCC(CNC(c2c(C)con2)=O)C1(C)C 58895,Cc1cccnc1C(F)(F)C(=O)NCCN(C(C1CC1C(F)F)=O)CCN(C)C 58896,N1(C(c2c(C)nc[nH]2)=O)CCC(C2CCN(C(C34CSC(C3)C4)=O)CC2)CC1 58897,c1(C(N2CCN(C(c3cnc(SC)s3)=O)C3C2C3)=O)cc2ncccn2n1 58898,N1(C(C)=O)CCC(NC(=O)CN(C)C(c2coc(C(C)C)n2)=O)CC1 58899,CCC(C)CC(C(=O)N(CC(C)(C)COC)C)NC(=O)C1=C(Cl)CCOC1 58900,N1(C(COc2cccc(C)c2C)=O)CCC(C2CC2NC(=O)CC(C)(C)F)CC1 58901,C12(C(N3CC(NC(COCCOC)=O)C3)=O)CC(c3ccccc3)(C1)C2F 58902,C1(C2CCN(C(=O)CCC3C(c4ccn(C)c4)C3)CC2)(C(=O)CCF)CCC1 58903,C1(CC(C)(C)C)CN(C(=O)COC2CCOCC2)CC1NC(c1ccoc1Cl)=O 58904,N1(C(COCCN(C)C)=O)CCCC1CN(C)C(c1csc(C2CCCO2)n1)=O 58905,C1(C(=O)NC(CCC(=O)N(C)CC)C)CC(=O)C12CCC2 58906,C1(OC)CC(C(N2CCC(c3ccco3)C2)=O)N(C(C2CS(=O)(=O)C2)=O)C1 58907,C1(CN(CC(=O)NC(c2ccccc2)CCC)C)CCCCC1C1CC1 58908,N1(C(C(CSC)OC)=O)CC(NC(=O)C(F)F)C(n2ccnn2)C1 58909,c1(C(=O)NCC(C)(C2CC2)NC(C(C)SC)=O)cc(Br)c(C)o1 58910,CC1(F)CN(C(c2cnc3[nH]ccc3n2)=O)CCN(C(C2CC3CCC2O3)=O)C1 58911,CCC(C)C(O)C(=O)N1CCCC(CC)(NC(=O)CC2CC3C=CC2CC3)C1 58912,C1(C(N2C(C)(COC)CC2)=O)CSCCN1C(c1ccc(CO)o1)=O 58913,N1(C(C(c2cc(C)oc2C)C)=O)CCC(CNC(c2nc(C)sc2C)=O)CC1C 58914,N1(C(CP(C)(C)=O)=O)CCOCC(CNC(C2CC(n3ccnn3)C2)=O)C1 58915,c1(SC)cccc(C(=O)NC2CCC(CNC(C3(C)COC3)=O)C2)c1Cl 58916,CC1(NC(c2nccnc2Cl)=O)CCN(Cc2ccccc2)CC1 58917,CC1CC(c2cn(-c3ccncc3)nn2)CCN1C(=O)CSC1CC1 58918,C(=O)(CCC(C)CN(C)C)NCc1occ(C(N(C2(C#C)CC2)C)=O)n1 58919,CC1CN(C(c2ccn(Cc3cccc(C(F)(F)F)c3F)n2)=O)CC(=O)N1 58920,CC1(C)CC(C(=O)NCCO)CN1CCCC1CCC1.C1(OC)CCCC1 58921,c1(OC)cc(F)c(NC(C2(C)CCN2C(=O)Cc2ncccn2)=O)c(F)c1 58922,C1(N(C(C(C)OCC(C)C)=O)C)CC2CCC(C1)N2C(c1cc2n(n1)CCC2)=O 58923,c1(NC(C2(F)CCN(Cc3nc(C)sc3)C2)=O)cncc(Br)c1C 58924,c1(C(N2C3CC(NC(C(C)OCC=C)=O)C2CC3)=O)ccc(C#N)c(C)c1 58925,N1(C(CN(C(C)=O)C)=O)CCCCC1C1CCN(C(=O)C(C)CC2CC2)CC1 58926,N1(C(C(F)=C(C)C)=O)CC(NC(=O)Cc2[nH]cnc2C)C(C2CC2)C1 58927,C1(NC(C2C(NC(C(C(C)O)N(C)C)=O)CC=CC2)=O)CCCC(O)C1O 58928,C12(C(N3CCC(CNC(C(C)SCC)=O)C3)=O)COCC1CS(=O)(=O)C2 58929,N1(C(c2ncn(CC)n2)=O)CCC(NC(c2cn(C)ccc2=O)=O)CC1C1CC1 58930,C12(C(N3CC4C(NC(c5cccc(C)c5F)=O)C4C3)=O)CCCCC1OCC2 58931,Cc1oc(C)c(CNC(=O)N(C)CCCSc2nc(-c3cccnc3)no2)c1C 58932,C(=O)(C#CC1CCCCO1)NC1CCC(NC(c2sc(C)c(Br)c2)=O)CC1 58933,c1(C(=O)NC2(CCNC(c3c(C)c(Cl)cnc3)=O)CC2)ccn2cncc2c1 58934,S(=O)(=O)(c1ccc(Br)cc1F)N1C2CCN(C(c3ncccc3Cl)=O)C2CCC1 58935,CCC(F)(F)CC(=O)NCC1CN(C(c2coc(C3CC3)n2)=O)CCCO1 58936,c1(C(N2C3C(N(C(C(C)P(C)(C)=O)=O)C)CC(C3)C2)=O)cc(=O)n2nccc2[nH]1 58937,CC(CC(=O)NCC(CNC(=O)C=CC=C(Cl)Cl)CO)c1cnn(C)c1 58938,c1(N2CC3CC(NC(C=C(C)c4ccco4)=O)C3C2)ncc2c(n1)CCCC2 58939,N1(C(C(CC(=C)C)OC)=O)CCCC(O)(CNC(=O)C(C)OCC)CC1 58940,c1(C(N2CCN(C(C3(CC)CC3(F)F)=O)CC2CO)=O)ccc2c(c1)CCC=C2 58941,C12CCCC(C1)C2.Cc1nc[nH]c1C(=O)NC1(C)CN(C(=O)CCC2CC2C)C1 58942,c1(C(=O)NC2C(NC(c3ccc(C(N)=O)cc3)=O)CCC2)cccc(O)c1F 58943,C12CS(=O)(=O)CC1CN2.c1(CNC(=O)CN(C2CCSC2)CCO)ccccc1 58944,C1(CNC(c2ncn(C(C)C)n2)=O)CC(C)CCN1C(=O)CP(C)(C)=O 58945,C(=O)(CC(C(F)(F)F)NC(=O)CC(C)C1CC1)NCCN(CCOC)C 58946,Cc1cc(C(=O)N(C2CN(C(=O)CCc3cnn(C)n3)C2)C)cn1C(C)C 58947,C1(C(N(C2CCCN(C(c3ccsc3)=O)CC2)C)=O)CC(F)(F)C12CCC2 58948,CCC(CN(C)C)CC(=O)NCC(CNC(c1ccc(N)c(F)n1)=O)S(C)(=O)=O 58949,c1(CNc2c(F)cc(C(F)(F)F)cn2)ccc2ncc(Br)cc2c1 58950,c1(C(CO)NC(C(C)C#N)=O)ccc(F)c(Cl)c1 58951,N1(C(CC=CC)=O)C2CCC1C1CC1(NC(C1COCCN1CC(F)(F)F)=O)C2 58952,C(=O)(C(C)(CO)NC(C1CC(n2cnnc2)C1)=O)OC 58953,C1(CC(=O)NCC(C2(O)CN(C(C(C=CC)O)=O)C2)(C)C)CCCC12CC2 58954,C(=O)(C(O)CC(=O)OC(C)(C)C)NCCCN(C(COCC#C)=O)C(C)C 58955,N1(C(C2(CC3CCC3)CC2)=O)CCCC(O)(CNC(C2(F)CCS(=O)(=O)C2)=O)C1 58956,c1(-c2cc(-c3nc(CCCCCC)nn3CCOC)ncc2)cc(F)cc(Cl)c1 58957,C=CCC(CC(F)F)NC(=O)C(COC)NC(=O)Cc1ccc[nH]1 58958,C1(N(C(=O)CC2CCCCN2C(=O)CC(C)N(C)C)C)CCCCCC1O 58959,N1(C(c2n(C)nc(O)c2)=O)CCS(=O)(=O)C(CCNC(=O)CC2(C(F)F)CC2)C1 58960,CCC(CC)(CCNC(c1nnn(-c2ccc(Cl)cc2F)c1C(F)F)=O)OC 58961,n1(CC)ccc(C(=O)NCCCCCCNC(c2csc3nnsc23)=O)cc1=O 58962,C1(C(N(CCC(=O)NCC(C#C)CC2CC2)CC=C)=O)C2CCCCCC12 58963,N1(C(c2n(CC=C)ccc2)=O)CC(C)OC2(CCN(C(=O)C(F)C(C)C)CC2)C1 58964,CCCC(C)(C)CC(=O)N1C2CCC1CN(C(C1(n3nccn3)CC1)=O)C2.C1(CC)CC1 58965,N1(C(C2(CNC(CCN(C)C)=O)CCCO2)=O)CCSC(C)(C)C1 58966,C1(OC)CCC12CC(C(=O)NC1CC1NC(c1c(C)noc1C(F)F)=O)C2 58967,c1(OCCC(=O)N(C2(O)CCN(C(C3(SCC)CC3)=O)C2)C)ccc(C)c(C)c1 58968,c1(OC)cc(C(N2CC3CC2CCC3NC(=O)CCS(N)(=O)=O)=O)c(O)c(Cl)c1 58969,C1(NC(C(C)N(C(c2cnn(CCO)c2)=O)CC)=O)CCCCCCC1 58970,c1(C(=O)NCC(CN(C(CCC(=O)NC)=O)C)O)ccc(OC)c(S(N)(=O)=O)c1 58971,C1(NC(c2c(OC)cncc2)=O)CCN(Cc2ccc(Br)[nH]2)CC1O 58972,C1(C(=O)NC(CNC(c2c(C)nn(CC(C)C)c2Cl)=O)(C)C)CN(CP(C)(C)=O)C1 58973,C#Cc1ccc(C(N2CCC3CN(C(=O)C(CCC)OCC)C3C2)=O)cc1C 58974,c1(C(N2CCCCC(NC(C(C)(C)c3cnsc3)=O)C2)=O)cn2c(n1)COCC2 58975,c1(C(=O)NCCC2(CNC(CCC(C)OC)=O)CC2)cnn2ccncc12 58976,c1(C(=O)NC2(CCNC(C(CC#C)C3CC3)=O)CC2)ccc(C)cc1C 58977,C1(CNC(C2CC(SC)C2)=O)CCCCN(C(c2c[nH]c(=N)s2)=O)C1 58978,C1(C(C)(C)C)(CNC(C2(C)CCCS2)=O)CCN(C(c2ccncc2)=O)C1 58979,C1(CNC(=O)NCC2CC(O)(C(F)(F)F)C2)(CO)CC2CC2C1 58980,CC(=O)CC(C)(C)CC(=O)N1CCCC1CCNC(=O)C#CC1CCCOC1 58981,CON(CC1CC1)C(=O)C(F)CC(C)(C)NC(c1cnc(O)c(C)c1)=O 58982,Cc1ccc(C(=O)NCC2CCC(NC(c3cnns3)=O)C2)cc1C 58983,N1(C(C=C)=O)CC(C)(C)CC1COC(C1CCC(C(F)(F)F)O1)=O 58984,C1(C2CC2)(C(=O)NC(CNC(C(C=C)O)=O)Cc2ccccc2)CCC1 58985,c1(C(N2CCN(C(C)=O)CC2c2cccc(F)c2)=O)cccc2ccn(C)c12 58986,Oc1c(CNCCc2cc(Cl)ccc2Cl)cc(Br)cc1Cl 58987,N1(C(C(CC2CCCC2)NC(c2cc(CC)oc2C)=O)=O)CCC2(CC1)CSC2 58988,C1(C(=O)NCCNC(c2cc(CC)no2)=O)CC1C1CCC1 58989,C=CCN=C(NCCc1nccc(C(F)F)n1)NCc1nc(C)cs1 58990,c1(C(=O)NCCOC2CCN(C(C3CC(C)N(C)C3)=O)C2)c(F)cc(F)cc1Cl 58991,c1(C(=O)OC)c(C)[nH]c(C(=O)NC2CC(N(C)C(C3C=CCC3)=O)C2)c1C 58992,N#CC1(CC(=O)NCC2CC2CNC(=O)CC2(CSC3CCOC3)CC2)CCC1 58993,Cc1cc(NC(=O)C(Cn2cncn2)NC(=O)CC2CSCCO2)cs1 58994,C1(OCC(=O)NC2CN(C(C)=O)C2)CCN(C(=O)Cc2ncc(Cl)s2)C1 58995,c1(C(C)OC(C(c2cn(CC)nc2)(F)F)=O)nc(O)c2ccc(Cl)cc2n1 58996,Cc1nocc1C(N1CCCC1CNC(=O)C=CC(=O)NCc1ccncc1)=O 58997,C(CC(C)CC)(C(=O)NCc1nc(C)c(C)s1)NC(CC(=O)NCC#C)=O 58998,C(C(COC)CC(=O)N1CCOC(C(=O)NCC2CCC(=O)NC2C)CC1)OC 58999,N1(C(C=CC(CC)C)=O)CC(C2CC2)(C(=O)N(C)Cc2ccc(SC)o2)C1 59000,C(=O)(C(CCC1CC1)NC(=O)C=CC1CC1)N(C1CSC1)C 59001,N1(C(C(CSC)O)=O)CC(F)CC1C(=O)NOCc1ccccc1O 59002,CC(C(=O)NCC1CCCCC1NC(C1(C#N)CCC1)=O)C1=CCCC1 59003,CCC(CC)CC(F)C(=O)N1CCC(CC(N2CCC3(C=CCO3)C2)=O)CC1 59004,c1(C2CN(C(=O)CNC(C3(c4nc[nH]n4)CC3)=O)C2)cccc(O)c1 59005,C1CCC2(CCC2)O1.c1(C2C(C3(c4n(C)nnn4)CN3)C2)ccc(I)cc1 59006,C(C(F)(C(=O)NC1(c2cccnc2)CC1)C(C)C)NC(C(C)C)=O 59007,CC(C)C(C(=O)N1CCC(CNC(=O)CNC(N)=O)C1C1CC1)NS(C)(=O)=O 59008,c1(C(=O)NC(C2(C(=O)N(C3COCC3O)C)CC2)C)cn(C)cn1 59009,Cc1cccc(C(=O)N(C2CCCCC2NC(C2OCCCO2)=O)C)c1 59010,N1(C(C(C2CCC2)OC)C(=O)NC2CCOC2)C2CCC1CC(=O)NC2 59011,C1(CC(=O)OC)CCC(NC(C2CN(C(c3ncccc3SC)=O)C2)=O)CC1 59012,N1(C(=O)CCSCc2ccccc2)CC2(CCN(C(=O)C3=CCCOCC3)C2)C1 59013,N1(C(c2ccn(CC)c2C)=O)CCN(C(c2ccc(O)c(C)c2)=O)CC1C 59014,CN(NC(=O)C(F)c1ccc(F)cc1)c1ncccn1 59015,c1(CNC(C(N2CC(C)C(F)(F)C2)c2nc(CC)[nH]n2)=O)ccc(F)c(F)c1 59016,c1(C(=O)NCCCN(C(CCOCC#C)=O)C)c(C)nc2sc(C)nn12 59017,c1(OC(C)=O)ccc(OCCC2CCCN(C(C)C)C2)cc1C 59018,C1(NC(C(C)OCc2ccccc2)=O)CC2CCC(C1F)N2C(C1(Br)CC1)=O 59019,C1(OCC)CC2(C1)CC2C(=O)NCCC(C)NC(=O)C(F)(F)COC 59020,c1(C(=O)NC(CNC(CSC)=O)(C)C2CC2)nc(O)[nH]c(=O)n1 59021,CCCCCC(O)C(=O)N1CCC2C(NC(=O)CN(c3ccccc3)C)C2C1 59022,c1(C(=O)NC(C(=O)NC(CC#C)C(=O)NC)CCSC)cccc(F)c1F 59023,n1(C(CC)C)ccc(=NC(=O)C(CC(N)=O)NC(c2cc(C(C)=O)c[nH]2)=O)[nH]1 59024,C1(NC(C2N(C)CC(O)C2)=O)C2CC3C(C2)C13C(N1CC(F)(C#N)C1)=O 59025,C1(CNC(C2(COC)CCOC2)=O)CCCCN(C(=O)CSc2nc[nH]n2)CC1 59026,c1(CC)ccc(F)c(C(=O)N(C2CCN(C(c3cn[nH]c3)=O)CC2)CCO)c1 59027,C1(OC)CC2CN(CC(c3ccccc3)Sc3ccc(F)c(F)c3)CCN2C1 59028,CCCCCC(=O)NCC(O)CN(C(=O)C(C1CCCOC1)OC)C 59029,Cc1nc(CNCC(F)(F)CCC(C)(C)C)oc1-c1ccccc1 59030,C1(C(=O)OC)(NC(=O)C(N2CCCNC2=O)Cc2ccccc2)CCCCC1 59031,C1(CNC(C(F)=CC)=O)CCCC1C(=O)NCCSC 59032,CC1CN(C(=O)CCC(C)(F)F)CCC1NCc1ncccn1 59033,C1(C(=O)NCCC2CC(F)(F)C2)(OC)CN(C(=O)CC2CCSC2)C1 59034,CC(C)C(CNC(=O)CC(O)CN(C)C)C(=O)NCCCSC(F)F 59035,CC1c2cccc(F)c2CCN1C(CCCCC1CCCC1)C(=O)NC(C)(C)C 59036,n1(CC(=O)NC(C)CN(C(=O)C=Cc2ccc(F)cc2)C)cnc2c1CCCC2 59037,CCC(CCOC)C(=O)NCc1cnn(C)c1C(=O)NCC1CC12CC2(F)F 59038,c1(CC(N2CC(=C(CNC(C)=O)F)C2)=O)cc(Cl)ccc1Cl 59039,c1(CN2CC(NC(C(C)Oc3ccccc3)=O)C(C#N)C2)cccc([N+](=O)[O-])c1 59040,NC(=O)CC(c1cn(C2CCC(NC(=O)C(C3CCCCC3)O)C2)nn1)C1CC1 59041,N1(C(C(C)(C)CF)=O)CC(CNC(c2ccncn2)=O)C(F)(F)C1 59042,Cc1cccc(CNC(C23CCC(NC(C4CCC(CO)O4)=O)(CC2)C3)=O)c1F 59043,c1(C(=O)NC(c2cn(Cc3cnoc3)nn2)C)ccoc1-c1ccccc1 59044,N1(C(CCCCSC)=O)CCC2(CC1)CC2C(=O)NC1(C)CC1(C)C 59045,CC1CCC(NC(C2(C(F)F)CC(F)(F)C2)=O)CN1C(=O)C=CCN(C)C 59046,CC#CCC(C(=O)O)NC(=O)C(c1ccc(Cl)c(F)c1)F 59047,c1(-c2ccc(N3CCCC(C=C)C3)c(N)c2)ccc(C#N)cc1F 59048,CC1CCC(C(=O)N(C(CNC(=O)CCCNC(=O)C(C)(C)C)C2CC2)C)C1 59049,C1(CN(C2CCN(Cc3ccnn3C)C2)C)CC(=O)N(CCc2ccccc2)C1 59050,Cc1cnc2c(C(=O)N(CCC(C)NC(=O)C(O)CN(C)C)C)cnn2c1 59051,C(C(F)(C(=O)NC1CCN2CCC1C2)C(C)C)NC(Cc1cn(CC)nc1)=O 59052,C1(NC(C=CCCC)=O)CC(C)(NC(=O)CNCCCC(C)NC(=O)OC)C1 59053,CCCC(C)(C)C(=O)NCCc1ocnc1CNC(=O)COc1ccc(Cl)c(C)c1 59054,N1(C(c2nc(CC)sc2)=O)CCCC(O)(CNC(c2ccnc(Cl)c2OC)=O)C1 59055,n1(CCC(=O)N(CCNC(C2CCC(C)O2)=O)CCOCCO)ncn(C)c1=O 59056,c1(C(=O)NCCC(C)NC(C(CSC)O)=O)scnc1C#N 59057,O=C(CS(=O)c1ccc(Cl)cc1)NCC1CCCN1C(=O)CC1CCCOC1 59058,c1(C(=O)OCCC(C(=O)OC)C2CCCCC2)csc2c1CCOC2 59059,C12(CNC(c3ccc(SC)o3)=O)CN(C(=O)C(C)SC(C)C)CC1CCO2 59060,c1(NC(C)=O)cnc2n1CCN(C(N1CC(O)(CN(C)C)C1)=O)C2 59061,Cn1nc(CC(=O)NC(CCN)C(F)F)cc1Cl 59062,c1(C(=O)NCCN(C(c2cc(C)cc(Cl)c2)=O)CC)ccc2nccnc2n1 59063,N1(C(c2nc(CC(C)C)sc2)=O)CCC(n2cc(CNC(=O)CO)nn2)CC1 59064,C1(NC(c2cc(F)cc(F)c2)=O)CC2CN(C(=O)CC3CCSCC3)CC12 59065,N1(C(C=C(COC)C)=O)CC2CCCC2(NC(c2nc(C(C)C)ncc2Cl)=O)C1 59066,C1(CNC(C(=Cc2cccs2)C)=O)(Nc2ncn(C(C)(C)C)n2)CCCCC1C 59067,c1(C(=O)NC2CCC(N(C(C(C)NC(CC)=O)=O)C)CC2)cc([N+](=O)[O-])ccn1 59068,CN=C1N=C2NC(=NCC(C(C)C)CN(C)C3CCCN2C3)N1.N(C)C.OC 59069,c1(C(N2CCCC(N(C(C(CC=CC)C)=O)CCF)C2)=O)cc(C)cc(C)c1O 59070,c1(C(=O)NCC(CC)NC(C2CCCC(F)C2)=O)c(OC)cccc1O 59071,c1(C(=O)NC(CNC(C(C2CCC2)OC)=O)C(C)(C)C)c(C)cc(C)nc1O 59072,C(=O)(C(O)CCCNC(=O)CC1(O)CCCOC1)N1CCC(C(C)OC)CC1 59073,c1(NC(C)Cc2ccc(CO)cc2)ccc(S(=O)(=O)NC2CSC(C)C2)cc1Br 59074,C(c1cc(Cl)cc(Cl)c1)=CC(=O)NCC(CNC(C1CC(CC)C1)=O)(C)O 59075,C12(C(=O)NCC3(C)ON=C(C)C3)CC(CN(C(=O)CCC(C)C)C1)C2 59076,CCC(CC)C(C)C(=O)N1CCOCC(NC(=O)Cn2cc(Cl)cn2)C1 59077,C(CC(C)C)(C(=O)NCC1CN(C(c2cccnc2O)=O)CCCO1)NC(C)=O 59078,C1(NC(COCCCCC)=O)CC2CCC1N2C(c1cnns1)=O 59079,C1(C(=O)NC(C2CCS(=O)(=O)C2)(C)C)CC2(CCC2=O)C1 59080,C(=O)(CCCC(=O)OC(C)(C)C)NC(C1CCN(C(CCCCOC)=O)CC1)(C)C 59081,Cc1ncc(C(N2C(C(=O)N(CCCCN(C)C)C)CCC23CC3)=O)c(C)n1 59082,C1(C(=O)NCCC2(C(=O)NCc3ncc(C)cn3)CC2)CC2CCC1CC2 59083,C(=O)(C1=CCN(C(C2CC2OC(C)=O)=O)C1)N1CCC(=C)CC1 59084,Cc1ncsc1C=CC(N1CCC(C(C)NC(C2C(C)(C)C2(F)F)=O)CC1)=O 59085,c1(C(N2CCOCC(NC(=O)CCCN3CCCC3)C2)=O)cn2ccncc2n1 59086,C(C)(CCC(=O)NC1CCN(C(=O)C(F)(F)c2cnn(C)c2)C1)SC 59087,C(=O)(CCCCN(C)C(C)C)NC(c1ccc(F)cc1)CNC(C(CC)=CC)=O 59088,C1(C(=O)NC(C2CCCC2)C#C)CN(C(=O)C(O)c2ccco2)CCC1(C)C 59089,CCC(COC)(CC)C(=O)NC1CN(C(=O)CCC2CC(OC)C2)CC1N(C)C 59090,C1(CC=C)(NC(=O)CCN2CCCCC2)CCN(C(C2(C(=O)NC)CC2)=O)C1 59091,C1(C2CCCCC2)(NCCC(C)N(C)Cc2ccccc2)CC1 59092,C1(NC(C(C)Cc2ccccc2)=O)CC12CC(NC(=O)CCCn1ccnn1)C2 59093,CCC(C)C(C)C(=O)N1CC(N(C(=O)CCc2c(C)nn(C(C)C)c2C)C)C1 59094,c1(C(N2CCC(CCNC(c3ccc(COC)[nH]3)=O)C2)=O)cc(N)c(O)c(F)c1 59095,N1(C(C2CCN(C(c3n(CC)ccn3)=O)C2C(C)C)=O)CC2(CCC2O)C1 59096,C1(NC(C(C)N(C(C)=O)CCO)=O)CCN(C(=O)CC2CCC(=O)N2)CC1C 59097,C(c1cccc(F)c1F)=CC(N1CC(NC(c2onc(C)c2C)=O)C(O)CC1)=O 59098,c1(C(N2CCC(N(C(=O)C(C)CC3CC3)CC#C)CC2)=O)ccc(=O)n(CC)n1 59099,CCS(=O)CC(=O)NCC(C)(C1CC1)NC(=O)CC1CC(C)(C)C1 59100,c1(C(C(=O)NCCCC(=O)NC)NC(=O)CSCC(N)=O)c(C)cccc1Br 59101,C1(C)(NC(C(n2cc(Br)cn2)C)=O)CCCN(C(C2(O)COC2)=O)C1 59102,c1(N(S(=O)(=O)c2cc(Br)cc(Br)c2)CC)ccc2c(c1)CCC(=O)N2 59103,C(=O)(C(C)CS(=O)(=O)c1ccc(F)cc1)NCC1=CCN(C(C=NOC)=O)CC1 59104,C1(C)(C(N(C)CC2CCN(C(c3ccon3)=O)C2)=O)CCCN1C 59105,CC(C)CC(O)CNc1nccc(N2CCN(CCN3CCOCC3)CC2)n1 59106,n1(CC)cc(Br)c(C(=O)NCC(O)CCNC(c2[nH]c(O)nc2C)=O)n1 59107,CC(CC(F)(F)F)C(=O)NC(CCF)C(=O)NCC1CCC(=O)O1 59108,c1(C(CC)C(=O)NC(C)(C)CCNC(=O)CSc2nc[nH]n2)cccc(Cl)c1 59109,N1(C(c2ncn(C)n2)=O)CC2CC(NC(=O)C=Cc3ccco3)CC(C2)C1 59110,C1(N(C(CN(CC#C)C(C2CCSC2)=O)=O)C)CCCOC1 59111,C12(C(=O)NC(C)C(=O)NC(C)(C)C)CC(CCO1)N(C(=O)C(C)N(C)C)C2 59112,C1(C(N2CC(C)(NC(c3cncc(-n4ccnc4)n3)=O)C2)=O)CCC2CC1CO2 59113,C1(CNC(C(C)OCC#C)=O)(CO)CC12CCN(C(=O)CC1CC=CC1)CC2 59114,Cc1nc(C(N2CCSCC2C(=O)NCc2ccncc2)=O)ccc1Br 59115,N1(C(c2c(SC)cnn2C)=O)CCC2(CCC2CNC(=O)C(F)(F)C(C)O)CC1 59116,C=CCC(C(=O)NC1CCCCN(C(=O)C(C)(C)C(=O)OCC)CC1)C(C)C 59117,c1(C(N2CCCN(C(c3nn(C)c(=O)cc3)=O)CC2)=O)ccc2ncn(C)c2n1 59118,CC1CCCc2cc(C(=O)NCCCNC(C3CCC4(CCC4)OC3)=O)nn21 59119,N1(C(CC(C)N(C)C)=O)Cc2nccn2CC(NC(=O)Cc2cnccc2Cl)C1 59120,N1(C(c2ccc(C)cc2C)C(=O)NCCOC)CC(C)OC2CCCCC12 59121,Cc1n[nH]c(C)c1CCCNC(=O)NCCc1coc(-c2ccccc2)n1 59122,C1(CCCNC(C=CCOC)=O)CCN(C(C2COCC2(C)C)=O)CC1 59123,c1(C(=O)NCC2CCN(C(c3cn(C)nc3Cl)=O)CC2)coc2ccc(F)cc12 59124,c1(C(N2C(CNC(C3CC34CC4)=O)C=CC2)=O)cc([N+](=O)[O-])ncc1Br 59125,c1(OC)ccc(Cl)c(CN2CCCC(C(=O)Nc3ncc(F)cc3Br)C2)c1 59126,c1(C(=O)NC2CCN(C(C3(C#N)CC4CC4C3)=O)CC2)ccnc2ccccc12 59127,N1(C(CNC(CNC(CCC(C)OC)=O)=O)=O)CC2(CCC2O)C1 59128,C1(CC(=O)N(CCCOCc2ccccc2)C)CCc2ccccc2C1 59129,C(C(CO)(CO)NC(=O)C(C)Cc1cnc[nH]1)N(C(C(C)OC)=O)C 59130,CCCCCC=CCCNC(c1[nH]ccc1CNC(=O)CC1CC(C)C1)=O 59131,N1(C(C(C(C)NC(C(=O)NCC)=O)C)=O)CC2CCC(C1)O2 59132,N1(C(CC2N(C(CCC(CC)C)=O)CC(F)C2)=O)CC(C2CC2(F)F)C1 59133,N1(C(CCOC(C)=O)=O)CC=CC1C(=O)NC(C)CN1CCCCC1 59134,N1(CC)C(=O)C(=Cc2cnc[nH]2)N(C)C=CC12CCCC2.c1ccc(F)cc1Br 59135,N1(C(C2CC2CC)=O)CC2(CCC(CNC(C3(C4CCCO4)CCC3)=O)O2)C1 59136,C1(C)(C(=O)NC(CC)C(=O)NO)CC12CCN(CCSc1ccccc1)CC2 59137,CC1CN(C(C2CCN(C)C2=O)=O)CC(C)CN1C(c1cc(O)cs1)=O 59138,CCCC(CCC)CC(=O)NCC(O)CNC(c1sccc1CC)=O 59139,c1(C(=O)NC(CNC(C2CC(OCC)C2)=O)(C)C)cc(Cl)c(Cl)cc1OC 59140,CN1CCC(C(=O)NCCC2(O)CCN(C(=O)CCC3CC3(C)C)C2)CC1 59141,c1(OC)cc(F)c(CNC(=O)Cc2cc(F)cc(F)c2)c(F)c1 59142,CC1(CNC(=O)C=CC(=O)NC2CC2)CCCN(C(=O)CC(F)(F)Cl)C1 59143,C(N=c1[nH]c(=NC2CC3CC4C(C3)C24)c2ncccc2[nH]1)c1nn(C)nc1Br 59144,O=C(C#CCNC(C1CCC(=O)O1)=O)NCCCOCC1CCC1 59145,S(=O)(=O)(c1ccc(=NCCn2cccnc2=O)[nH]c1)NC(c1ccccc1Br)C 59146,C(=O)(C1=CC2CCC(C1)C2)NC1C(NC(c2ccc(C)c(C#N)c2)=O)C1 59147,c1(C(=O)NCCC2N(C(C3CCN(C)C3)=O)CC(F)(F)C2)cn(C)c(=O)nc1O 59148,c1(CC)ccc(C(=O)Nc2ccc(NC(=O)NC3(O)CN(CC)C3)cc2)cc1 59149,C1(NC(c2cc3ccsc3[nH]2)=O)CC2CC(C1)N(C(C1Cc3nccn3C1)=O)C2 59150,C(c1ccc(S(C)(=O)=O)o1)=CC(=O)NC1CC(CCNC(C(C(C=C)C)C)=O)C1 59151,c1(C(=O)NC2CC(C(=O)Nc3ccc(C4CC4)cc3)C2)ccc(Br)c(Cl)n1 59152,C(=O)(C(CC)C(C)(C)CC)NC1CCC(CNC(c2ccc(C#C)o2)=O)CC1 59153,C1(NC(CC(C)n2cccn2)=O)C2CCC1CN(C(=O)C(=O)NCC(F)F)C2 59154,C1(C(=O)NC(CCCNC(Cc2cc(C)ns2)=O)C)CCN(C)C(=O)C1 59155,Cc1c(C(=O)NCC#CCNC(=O)CC2CCCC2(F)F)sc2ccccc12 59156,c1(C(c2ccc(OC)cc2OC)N(CC(=C)C)C=O)ncc(Cl)cc1Cl 59157,C12(NC(c3cccc(Cl)c3)=O)CCCCC1N(C(c1ccncc1)=O)CC2 59158,O=[N+]([O-])c1cncc(-n2ccc(Nc3ncnc4ccsc34)n2)c1 59159,Cn1nc(Cl)c(C(=O)NC2CCN(C(=O)CCC(C)(C)C)C(C3CC3)C2)c1Cl 59160,c1(CNC(C=CCC)=O)csc(CNC(c2cc(F)cs2)=O)n1 59161,c1(N2CCC(NC(C(C3CC3)OCC)=O)(CF)C2)ncc(Cl)c(O)n1 59162,N1(C(COC)=O)CCC2(NC(c3cncc(C(=O)OC)c3)=O)CC2C1 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59180,c1(-c2cn(CC3CC(NC(C4CC(=O)C4)=O)C3)nn2)cc(F)ncc1Cl 59181,C1(NC(c2c(C)ncs2)=O)CCCCC1NC(c1ccc(C(C)(C)C)o1)=O 59182,c1(NCC)ncc(C(=O)N(C)CCN(C(=O)C(C2(O)CCCC2)F)C)cc1Cl 59183,n1(CC)cnc(C(=O)NC2CCC2NC(C2(F)CC2)=O)n1 59184,C12(CNC(CNC(=O)C3CC3)=O)CCCCC1CN(C(=O)C1=C(Cl)CCOC1)C2 59185,S(=O)(=O)(c1ccc(NC2CCCC3(C2)OCCO3)c(C#N)c1)NCCC(C)F 59186,c1(CNCC2C(C)CC2)oc(C(=O)O)cc1Br 59187,c1(C(C(=O)NC2CCC2)N(CCC2=CCCCC2)C)cc2cc(Cl)ncc2o1 59188,N1(C(c2c(OCC)nsc2)C(=O)Nc2ccccc2)CCN(CCC(F)F)CC1 59189,n1(CC(N2C3CC(CNC(C(CC=CC)C)=O)C2CC3)=O)cnc2ccccc12 59190,c1(NC(Cc2c(C)nccc2)=O)cc(Br)c(F)cc1C#N 59191,C(C(CC(C)C)C(=O)NCC(C)(C)C1(O)CCC1)NC(C(CCOC)C)=O 59192,C(=O)(C(O)C(C(C)C)OC)N1CC(C(C(NOCCCC)=O)F)(O)C1 59193,N1(C(c2ccc(OC)nc2)=O)CCC(C)C(NC(C2(OC)CCSC2)=O)C1 59194,CCCCCCC(C)C(=O)N1C2CCC1CC(N(C)C(c1nc(C)oc1C)=O)C2 59195,c1(Cc2nc(CC(C)OC)nn2-c2ccn(C)n2)ccc(Cl)c(Br)c1 59196,N1(C(CC2C(C)C2)=O)CC2CC2(NC(c2ccc(OCC3CC3)nc2)=O)C1 59197,C(C(CC1CCCC1)C(=O)NC1CCC(O)C1)NC(=O)CC1(CO)CC1 59198,c1(C(N2CCC(CNC(C3C(C)OCC3)=O)C2)=O)cnn2ccn(C)c12 59199,C12(C(N(CCCC)C)=O)CCC(n3cc(C4CCCO4)nn3)(CC1)C2 59200,CCS(=O)CC(=O)N(CC(C)CNC(=O)CCCSC(C)(C)C)C 59201,CC1CN(C(=O)Cc2ccnn2C2CCOCC2)CC1NC(=O)Cn1ncnn1 59202,c1(N(C)C)cc(-c2ccc(C(=O)NCC3COCCO3)nn2)cc(C#N)c1 59203,C(CC(C(=O)NC(COC)CO)NC(C1CC(OC)C1)=O)SC 59204,S(=O)(=O)(c1cccc(N(C)Cc2scnc2C)n1)N1CCC(OCC=C)C1 59205,c1(C(=O)NC2CC(CCNC(=O)CN3C(=O)CNC3=O)C2)nnn2c1CCCC2 59206,C(N=c1[nH]c(=N)[nH]c(=NCCS(=O)(=O)CCO)[nH]1)C1(C=C)CCOCC1 59207,S(=O)(=O)(CCC(F)(F)F)N1CC(CNC(c2cnc(Cl)c(F)c2)=O)NCC1 59208,N1(Cc2cccc(OC)c2F)Cc2ccccc2C1C(=O)N1CCOC(CO)C1 59209,c1(C(=O)NC2CN(C(C3N(CCC)CCCC3)=O)CC2C)cc(C)c(Cl)cn1 59210,c1(CCCC)cc(C(=O)NCC2(NC(=O)C=Cc3cocn3)CCOC2)c(C)o1 59211,c1(OC)ccc2occ(C(=O)NC3CCCCC3CNC(=O)C=CC3CC3)c2c1 59212,C1(C(=O)NCCN(C2CCCC2)C(C23CCC2C3)=O)(CC)CCCCC1 59213,C(=O)(CCC(=O)NCC(C)(C1CCC1)NC(C1CCC12CCC2)=O)N(CC)CC 59214,c1(C(=O)NCCN(C(=O)C(F)(F)CO)CCC)ccc(=O)n2c1COCC2 59215,c1(C(=O)NCCC(C)N(C(Cc2cc(C)no2)=O)C)c(C(F)F)cnn1C 59216,C(C(C(=O)NCC(C)(O)CN(C)C)N(C)C)NC(C(C)NC(=O)CC)=O 59217,N1(C(CS(=O)(=O)NCC)=O)CCCC12CCN(C(c1ccccc1C(C)O)=O)C2 59218,C(=O)(CC(F)(F)CC)N1CCC(CC)C1CNC(c1cccc(=O)o1)=O 59219,c1(C(N2CC(NC(C(C(C)C)(C)C)=O)C(C(F)(F)F)C2)=O)ccc2nccn2n1 59220,C1(CNC(N2CC(n3cc(I)cn3)(CC(=O)OC)C2)=O)CC(C(F)(F)F)=NO1 59221,C12(C(=O)NC3C(NC(c4cccc(OC)n4)=O)CCC3)CCCCC(OC)(C1)C2 59222,C1(C(=O)NC2CCC(C(C)C)CC2)(CC)CCCN1C(=O)C(C1CCCCC1)O 59223,N1(C(C(C)N(C(=O)CC2(N(C)C)CC2)CCC)=O)CCCC(N(C)C)CC1 59224,C(=O)(CCC(F)(F)F)NC1C=CCN(C(C(CC#C)C2CC2)=O)C1 59225,C1(NC(C2C3(CC3)C23CC3)=O)CCN(C(=O)CN2CCOC2=O)CC(O)C1 59226,N1(C(CN(CCOC)C)=O)C2CCC(C2)C1CNC(=O)Cn1nc(C)oc1=O 59227,C12(CNCC3(N)CCC3)CC3CC(CC(C3)C1)C2 59228,C1(NC(c2nc(CCC)sc2)=O)CN(C(=O)COc2cccnc2)CC(C)(C)C1 59229,Cc1ccc(Br)c(C(N2CCC3(NC(=O)CCc4ncc[nH]4)CC3C2)=O)n1 59230,C(=O)(C1=NOC2COCC12)N1C(C(=O)NCCC2=CCOCC2)C=CC1 59231,Cn1nc(C(N2CCC(C(N3CC(c4ccccc4)C3)=O)C23CC3)=O)cc1C#N 59232,C(=O)(C(C)(C)CNC(C1CC(C)N1C(=O)CCc1cnco1)=O)OC 59233,N1(C(c2cc(CC)c(CC)o2)=O)CC(C2CN(C(=O)C(C)(O)CC)C2)C1 59234,c1(C(=O)NC2CN(C(CC3CC(CC)C3)=O)CC2C)c(C)nn(C(C)(C)C)c1C 59235,C(=O)(C1=NOCC1)N(CC(CNC(C(CSC)OC)=O)(C)C)C 59236,C(c1ccc(Cl)cc1)=CC(=O)NCC(CN(C(CC(=O)N(C)C)=O)C)(C)C 59237,C(CCCCC(=O)NC(CC1CC1)CO)NC(c1cc(OC)ns1)=O 59238,Cc1cc(C(N2CCC3(CC2)CC3NC(C2CCCC2)=O)=O)c2c(C)noc2n1 59239,C1(NC(CCC=C)=O)CN(C(=O)C(C)CN(C)C)CC1OCC 59240,Cn1c(O)nc2cc(C(N3CCC(CCNC(=O)CCCC#N)C3)=O)ccc12 59241,Cc1ccc(C)n1CC(N1CCCC1CCC(N1CCCC(F)C1)=O)=O 59242,C12(C)CCC(O1)N2.C(CC(=O)N(CCCN(C(=O)COC)C)C)OCCOCC 59243,c1(N2CC3CC(C)(C)C3C2)nc(=NCCc2cccc(F)c2)[nH]c2c1COCC2 59244,c1(C(=O)NC2C(NC(CN(C(=O)OC)C)=O)C2)cc2n(n1)CCO2 59245,C(=O)(C(c1ccccc1)=CC(C)(C)C)NC12C(CN(C(COCCC=C)=O)C1)C2 59246,c1(N(CCCN2CCOCC2)Cc2ccc(C)o2)ccc(F)cc1C#N 59247,C1(C(=O)NCCC(=O)NC(N)=O)CC(C)N1C(c1ncn(C)n1)=O 59248,CC(CC(N)=O)C(=O)NC1CCCC1NC(c1cc(N(C)C)ccn1)=O 59249,Cc1ccc(Cl)cc1-c1cn(CCCNC(=O)CCNC(N)=O)nn1 59250,c1(C(N2C(CC=C)CCCC2)C(=O)NC2CCCCCC2)c(C)cccc1C 59251,N1(C2CCN(C(CCCOCC=C)=O)C2)CCN(C(c2ccc(Br)o2)=O)CC1 59252,C(=O)(C(F)C(C)(F)F)NC(COCC=C)C(=O)OC 59253,C12(NC(c3nc(C(C)C)oc3)=O)CCCC1CN(C(=O)CN1CC3CC3C1)C2 59254,c1(SC)nccnc1C(N1CC(NC(c2c[nH]c(=O)cn2)=O)C1)=O 59255,S(=O)(=O)(c1cccc(F)c1Cl)NCC1CC[Si](C)(C)C1 59256,c1(C(N2C(CNC(c3cc(C)sc3)=O)C(C)CCC2)=O)ccc2c(n1)CCCC2 59257,c1(CN2C(C(=O)Nc3c(C(C)=O)cccn3)CC3CC32)c(C)cc(Br)cc1C 59258,c1(C(=O)C(=O)NC2CC(CF)C2)ccc(Br)cc1F 59259,c1(C(N2CC(NC(c3ccco3)=O)C(F)C2)=O)ccc(Cl)c(F)c1F 59260,c1(COC(C)C(=O)N(C)CC2CCS2(=O)=O)cn(CCCC(=O)O)nn1 59261,C(=O)(CC1CCc2ccc(O)cc21)N1CCC(=CCNC(COCC=C)=O)CC1 59262,c1(OC(C)C)ncc(C(=O)NC(C)CN(C)C(C2(C)CCCC2)=O)cc1Cl 59263,C(C#Cc1ncccn1)N1CCC(N(CC(CC)C)C)C1 59264,C(CCC1CC1)(C(=O)NC(c1ncn(C)n1)C)NC(C(n1c(C)ncc1)C)=O 59265,CCC(C)CC(C(=O)OC)NC(C12CC(C)(C1)OC2CN)=O 59266,C=C(C)CC(C(=O)N1CCC(CCCC)C1)NC(=O)C(C1CCOCC1)F 59267,c1(CC(=O)NCCN(C(=O)CN2CCCC2CO)CCOC)nonc1C 59268,N1(C(C2CN(CC(F)(F)F)C2)=O)CCCC(CC(=O)Nc2cc(C)no2)C1 59269,C1(C(=O)OCc2cccc(CC)c2)CCCCN(C(C2CCCN(C)C2)=O)C1=O 59270,C1(C(N2C(CCC(C)(C)NC(C(C=C)C)=O)CCCC2)=O)CCC(=O)N(C)C1 59271,C(=O)(C1=NN(C)C(=O)CC1)N1CCC(N(C(c2c(C)nns2)=O)C)C1 59272,N1(C(CCC=CC)=O)CCC(NC(=O)C=Cc2cccc(OC)c2)C(CO)C1 59273,c1(C(N2CCC(C(=O)OC)C2C)=O)n[nH]c2c1CN(C(=O)CCC1OCCO1)C2 59274,N1(C(c2coc(C3CC3)n2)C(=O)NCCOC)CCCN(CCC#N)CC1 59275,c1(C(=O)NC(CC)CN(C)C(C2CCOC(C)(C)C2)=O)ccc(=O)n2c1CCC2 59276,N1(Cc2c(OC)cccc2)CCC2(CC1)CC2C(N1CCCC1C(C)C)=O 59277,N1(C(C2N(CCCN=[N+]=[N-])CCCC2)=O)CC(C2CCCOC2)C1 59278,Cc1occc1C1CC1C(=O)NCCNC(=O)C(C)n1cccn1 59279,C1(NC(c2c(C)sc(Br)c2)=O)CC2CCCC(C1)N2C(C1CC1(F)F)=O 59280,C12(CNC(CCC(=O)N(C)C)=O)CCC1CCN2C(=O)COC1(C)CCCC1 59281,Cc1ccc(C(=O)NCCC(=O)NC2CCCN(C(C3(CO)CC3)=O)C2)c(O)c1 59282,Cc1nc(C(=O)NC2CCCC2(C)CN(C(=O)C(O)CC(C)C)C)cc(O)n1 59283,N1(C(c2c(C)nc[nH]2)=O)CCC2(CCCN(C(C3CCC4CC34)=O)C2)C1 59284,N1(C(CCC=C)=O)CCSCC1C(=O)N(CC(O)COCC)C 59285,N1(C(c2[nH]cc(C(N)=O)c2)=O)CCN(C(C2CC3CCCC3C2)=O)C(CO)C1 59286,C(CS(=O)(=O)c1ccc(C(=O)NC2CC2NC(=O)CCSC)cc1)OC 59287,C(C)(CCC(C)(C)C)NC(c1c(-c2cn(C(C)C)nc2)nn(C)c1)C1CC1 59288,C1(C(=O)NC2C(CC=C)COC2)CCC2(CC2)N1C(=O)CC1(C)CC1 59289,N1(C(C2N(CC)CC2)=O)CC(C)CN(C(c2cnoc2-c2cnccn2)=O)CC1C 59290,CC1=C(C(=O)NCC2CCCN(C(c3coc(C(C)C)n3)=O)C2)COCC1 59291,C1(C(C)NC(c2nc(Cl)cs2)=O)CCCN(C(=O)CC23CCC(CC2)C3)C1 59292,c1(OCC)cc(Br)c(NC(=O)C=Cc2ccc(C)nc2)c(Br)c1 59293,N1(C(C2C(CC)CCO2)=O)CCC(C(=O)NC(CN(C)C)C(C)(C)C)C12CCC2 59294,C(=O)(C1=CC2C=CC(C1)C2)N(C(C(=O)N(C(CCC=C)C)C)C)C 59295,Cc1nc(CC(C)C)c(C(=O)NCC2C3CN(C(c4ccc(Cl)cn4)=O)CC23)s1 59296,C1(C(F)(F)F)(C(=O)NCC=CCNC(=O)Cn2cnnn2)OC2CCC1C2 59297,c1(SC)ncc(C(=O)NCCOC2CN(C(C3CCCSC3)=O)C2)s1 59298,N1(CC=C(C)C)CCC2CN(Oc3ccc(C(=O)OCC)cc3)CC12 59299,c1(C(=O)NCC2(F)CC(NC(C(C)NC(C)=O)=O)C2)ccc(C)c(S(C)(=O)=O)c1 59300,N1(C(CC(C)N(C)C)=O)CCCCC1CCC(=O)NCC=C(Cl)Cl 59301,c1(C(N2CCc3ccccc3C2)=O)ccc2nnc(S)n2c1 59302,C1(NC(c2ncn(C(C)C)n2)=O)CN(C(C2CCCCS2)=O)CCC1(C)C 59303,C1(NC(C=Cc2c(OC)cccc2)=O)C2CCN(C(=O)C3=CCCOC3)CCC12 59304,C1(C(N(C2CCC2)CC#C)=O)CC(O)C(O)CC1CNC(C1CCCNC1=O)=O 59305,c1(NC(C2CC(O)(CNC(c3cocn3)=O)C2)=O)ccc(Cl)cc1O 59306,N1(C(c2n(CC)nnc2)=O)CCC2(NC(=O)Cc3cc(Cl)sc3Cl)CC2C1 59307,N(C(=NCC1CCN(C)C1=O)NC1CCOCC1)CC1(NCC=C(C)C)CCOC1 59308,C1(NC(CC2CCC(=O)NC2)=O)CCN(C(=O)CC2C=CCCC2)C12CCC2 59309,C#CCCC(C(=O)NC(CCC)C(=O)NC)NC(=O)C(F)C(F)(F)F 59310,N1(C(C2(C)CC=CCC2)=O)CCC2(CC(C(=O)N3CCCCC3C(N)=O)=NO2)C1 59311,C1(C(N(CCNC(CCc2cn(C)nc2)=O)CC2CC2)=O)CCc2nnnn2C1 59312,c1(C(N2CCC(O)C2)=O)cnc2c(-c3ccc4[nH]ccc4c3)cccc2c1 59313,C1(=CC(=O)NCC(CC)NC(c2ccc(C(=O)OC)[nH]2)=O)CC2CCC(C1)N2C 59314,C1(NC(C2CCN(C)C2)=O)CC2(C1)CC1(CC(NC(C3(C)CC3(F)F)=O)C1)C2 59315,C(=O)(C1=Cc2ccccc2C1)N1C(CC)C(NC(=O)C(F)(COC)C(C)C)CC1 59316,N1(C(C2CCCC3(CC3)C2)=O)CCC2(CC1)CN(C(=O)C(O)C1CCC1)C2 59317,c1(OC)cc(-c2ccc(F)cc2F)c(OC)cc1CN1CCCC(N(C)C)C1 59318,C1(NC(c2ccc(CN(CCC)C)o2)=O)(CF)CCN(C(C2CC(C)(F)C2)=O)C1 59319,C#CCC(C)(C(=O)NCC(C)C)NC(=O)C(CN(C)C)N(C)C 59320,C(=O)(C1=CCCOCC1)N1CCN(C(C(C)NC(C)=O)=O)C(CS(C)(=O)=O)C1 59321,CC1CCN(C(c2nonc2N)=O)CC1NC(c1cn(C)c(=O)cn1)=O 59322,N1(C(C2C(C(C)C)C2)=O)CC2(CCN(C(=O)CC(C)(C)C#N)CC2)CC1C 59323,N1(CC(=O)NC2CN(C(C3(CO)CCCCO3)=O)CC2O)CCS(=O)(=O)CC1 59324,C1(OC)(CNC(C2(C)CC=CCO2)=O)CCN(C(c2nccnc2C)=O)C1 59325,c1(C(=O)NCC2(OC)CN(c3cc(C(=O)OC)ncn3)C2)cc(F)ccc1F 59326,C1(C)(C(N(C)Cc2cncs2)=O)CCN(C(c2cc(CO)n(C)n2)=O)C1 59327,C1(C(N2CC(C)(NC(C(C)N(C)C)=O)C2)=O)CCCCN1Cc1ccccc1 59328,c1(OCC)ccc2cc1NC(=O)CCNC(=O)N2.c1(COC)nocc1CC.OC 59329,C1(OC)C(NC(C2OCCC2CNC(=O)CC2CC2)=O)CC1O 59330,C1(C(=O)Nc2nccnc2CC)COCCN(CC2(C#C)CCCC2)C1 59331,C1(NC(CCc2c(C)cccn2)=O)C(C)CCN(C(c2ccc(C#N)s2)=O)C1C 59332,C12(C(N3CC(CC)OCCC3)=O)CCC(CC1)N(C(c1ncncc1Cl)=O)C2 59333,c1(C(=O)NC2C(CC(=O)NCCCCC)CCC2)cnc(C)cn1 59334,C1(C(C)OC(c2ccc(C(CCC)=O)cc2)=O)NC(=O)CNC1=O 59335,CC(C)CC(C(=O)NC1CC1(C)C(F)F)NC(c1cnn[nH]1)=O 59336,O=C1CCCC(CC(=O)N(C2CCC2)Cc2cn(CCCC(=O)O)nn2)C1 59337,C1(CC(=O)NCC2(CN(C(=O)C(F)CC3CCC3)C)CC2)CC(F)(F)C1 59338,N1(C2C(C)OCC2)CCN(C(c2ccc(CNc3cccnc3N)cc2)=O)CC1 59339,c1(C(N2CC(CC(=O)NC3(C(=O)OCC)CCCC3)C2)=O)ccncc1Br 59340,Cc1nc(C(=O)NC2C3CCN(C(=O)CSC4CCS(=O)(=O)C4)C23)cc(O)n1 59341,c1(C(N2C3(CNC(CC(C)C(F)F)=O)CC(CO)(C2)C3)=O)ccc2nn[nH]c2c1 59342,c1(C(=O)NCC2CC(F)(CNC(C=CC(=O)OCC)=O)C2)cc2sc(F)cc2[nH]1 59343,Cc1cc(Cl)c(C(N2CCCC2CN(C(=O)C(C)CC(C)C)C)=O)cc1[N+](=O)[O-] 59344,c1(OCC(N2CC(NC(CC(=C)Br)=O)C3C2C3)=O)ccc2c(c1)CCC2=O 59345,N1(C(C(N2CCN(C)CC2)C)=O)CCN(C(c2ccc(N)c(N)n2)=O)C(C)C1 59346,c1(-c2cnc(NC(c3ccc(OC)cc3F)=O)c(C)c2)cnc(C#N)c(F)c1 59347,C1(NC(c2n(CC)ncc2)=O)CCN(C(c2ccc(CO)cc2)=O)CCC1CO 59348,C(CC(=O)N1CC2(CC(O)C2)C1)(C(F)(F)F)NC(=O)C=Cc1ccco1 59349,C1(NC(C2N(C(c3n(CC)nc(C)c3)=O)CCCC2)=O)CCC(C2CC2)C1 59350,C12(NC(c3cn(C=C)nc3)=O)CCC(C(N3CC4CCC3C4)=O)(CC1)CC2 59351,N1(C(c2ccc(OC)nn2)=O)CC(C)C(C)(C(=O)NC2(C)CCCCCC2)C1 59352,C12(CNC(C(CC)C)=O)CC(NC(c3cocc3Br)=O)(C1)C1(CCC1)O2 59353,C(=O)(C=C1SCC(=O)N1C)N(C1CCCC(NC(COCC#C)=O)C1)C 59354,C1(C(=O)NCc2c(CC)nco2)(C(=O)N(C2CSC2)CCN(C)C)CCCCC1 59355,C12(C(N3CC(O)(CCC)C3)=O)CC1CCN2C(c1ccn(C2CC2)n1)=O 59356,CC1CCc2c(C(N3CC(C)(C)CC3CNC(=O)CC3CC34CC4)=O)csc2C1 59357,C1(CCC)CN(C(=O)CC(C)COC)CCN1C(c1cn(C)nn1)=O 59358,c1(OC)cc(C(N2CC(NC(=O)CCc3n[nH]c(=N)s3)CC(O)C2)=O)cc(C)c1 59359,C=CCC(CC(F)F)NC(c1ccc(F)c(C)c1)C 59360,N1(C(c2n(CC)cc(Cl)c2)=O)CCCC(O)(CNC(C2C(C)(C)C2(F)F)=O)CC1 59361,c1(NC(CC2(C#N)CCNC2)=O)cccc2c1OCCC(=O)N2 59362,N1(CC)N=C(C(=O)NCC2C=CC(NC(c3ncc(Cl)cc3Cl)=O)C2)CCC1=O 59363,C(CCCCC(=O)N1CCN(C(c2cc(C(F)(F)F)c[nH]2)=O)C(C)C1)=CC 59364,N1(C(C(C)P(C)(C)=O)=O)CCOC2(C1)CN(C(C1CC13CC(O)C3)=O)C2 59365,C1(NC(C2Cc3nncn3C2)=O)CN(C(c2ccsc2)=O)CC2(CC2)C1 59366,c1(CNC(c2n(CCOCC)nnn2)C2CC=CCC2)ccc(F)c(C)c1Cl 59367,C1(OC)CCN(C(c2cc(CF)on2)=O)C1CNC(=O)OC(C)(C)C 59368,C(=O)(C1CCCc2sc(=N)[nH]c21)NCC(CCCC)NC(=O)CC(C)C 59369,C(C(=O)NCC1(CNC(=O)CCNC(=O)C(C)(C)C)CC1(F)F)(C(C)C)SC 59370,Cc1cc(Cl)c(C(=O)NCCC2CCCN(C(=O)COCc3nc(C)no3)C2)s1 59371,c1(C(N2C3CCN(C(c4c(CC)nc[nH]4)=O)CC3C2)=O)cn2ccc(F)cc2n1 59372,c1(C(N2CCN(C(C3CCN3CC(F)(F)F)=O)CC2)=O)cc(F)cc(Cl)c1 59373,c1(C(N2CCN(C(c3csc(C)c3C)=O)CC2C2CC2)=O)nc[nH]c2nccc1-2 59374,C(=O)(CCC(C)CC)N1CCC(CC=C)(C(N2CC(CS(C)=O)C2)=O)C1 59375,C1(CC(=O)NC(C)CNC(c2c[nH]nc2C(F)F)=O)CCCC(C2CC2)O1 59376,O(P(C)(=O)CNC(C1CC=CCN1C(=O)CC1CCCOCC1)=O)CC 59377,CCCCCCCCN(CC(=O)Nc1cc(N)nc(Cl)c1)CC(=O)OC 59378,N1(C(CC(N(C(C2CCC2)=O)Cc2cccc(C)c2)SC)=O)CCCN(CC)CC1 59379,C12(CNC(c3c(C)nsc3)=O)CCCC1N(C(=O)C(C)C1CCOC1)CCC2 59380,C1(CN(C(C(C=CC)O)=O)C)CN(C(=O)CC(CC)c2ccccc2)CCO1 59381,N1(C(C(=O)NC2CC(C(=O)OC)C2)CCC2CC2C)CCCC2(CCCOC2)C1 59382,c1(C(N(CCNC(C(CC)(CC)OC)=O)CC2CC2)=O)cnc2cc[nH]c2c1 59383,C1(CNC(c2nc(COC)oc2)=O)CCN(C(C2CC3(CC3)C2)=O)CC1O 59384,C1(C(=O)Nc2cn(CC=C)nc2)CSCCN1C(c1c[nH]nc1C)=O 59385,C(=O)(C(C(C)(C)C)NC(N)=O)NC1C(CNC(c2c(C)cno2)=O)C1 59386,CCC(C(=O)OC)C(=O)NC1CC2(C1)CN(C(=O)CSc1nncn1C(C)C)C2 59387,Cc1ccc(C(=O)NCC2CN(C(C3CCC3C(C)(C)C)=O)CCO2)c(F)c1Cl 59388,C(=O)(CCCCNC(C1C(NC(=O)CC2CC(C)(C)CO2)C1(C)C)=O)OCC 59389,c1(C(=O)NC2CCC(NC(c3ccnn3CC3CC3)=O)C2)ccn2ccnc2c1 59390,C1(CN(C(C2CC(C(F)F)(OC)C2)=O)C)CCN(C(C2CC(O)C2)=O)CC1 59391,C(N=c1cc(CC)nc[nH]1)C1(NC(C(CC)NC2CCCC2)=O)CCCCC1C 59392,C1(C(=O)NC2CC(OC)CN(C(=O)C(C)(C)C#N)C2)CS(=O)(=O)CC(=O)N1 59393,N1(C(C=CCOC)=O)CC(O)CC1C(N1CCCC1C1(C)CC1)=O 59394,c1(CNC(C2CC(c3ccon3)C2)=O)ccccc1CNC(C1CCCCO1)=O 59395,N1(C(c2cnc(CC)o2)=O)CCC(CC)C1CNC(c1ccsn1)=O 59396,C1(Br)(C(=O)NCCOCCN(C(C2(C)C(C)C2)=O)C)CC1(F)F 59397,N1(C(c2cn(C)nc2Cl)=O)CC2CC(C1)C(CO)C2NC(c1cccc[n+]1[O-])=O 59398,N1(C(CC)=O)CCC(C)(C(=O)OCC)CC1=O.C(C(C(C)C)N1CCCC1=O)O 59399,c1(C(CC)CN(C2CC2)C(c2nc[nH]n2)C)ccccc1 59400,CCCC(C)CC(=O)NC1COCCN(C(c2c(C)cccc2N)=O)C1 59401,CC1(C(=O)Nc2nnco2)CCN(Cc2cccc(I)c2F)CC1 59402,N1(C(C(CC)F)=O)CCC(N(C)C(c2cc(-c3ccoc3)[nH]n2)=O)C2(CC2)C1 59403,CC(C)CC(O)C(=O)NC1CN(C(c2cccc(SC(F)(F)F)n2)=O)CC1C 59404,CC1CC(N=c2c(Br)c[nH]cc2[N+](=O)[O-])CN1C(c1nc[nH]c2nccc1-2)=O 59405,C(CC(C)CCNC(c1cc(C(C)CC)no1)=O)NC(CCCOCC)=O 59406,c1(OC)ccc(CNC(=O)COOC)c(Cc2cn(C3CCOCC3O)nn2)c1 59407,C(=O)(C(CCOCC)NC(=O)C(C)C1CCCC1)N(CC=C)CCOC 59408,CC1(C)CCCC(CS(N2CCC(N3CCCCCC3)CC2)(=O)=O)O1 59409,c1(C(=O)NCC(C)(C2CC2)NC(CC(C)OC)=O)c(Cl)c2ccccc2n1C 59410,C1(N(C(C2C(SC)CCC2)=O)C)CCN(C(c2cnn(C3CC3)c2C)=O)CC1 59411,C(=O)(C(C)CC(F)F)NC1C(NC(CCc2cccc(C)c2)=O)CCCC1 59412,c1(C(=O)NCCCN(C(=O)Cc2cnsc2)C(C)C)cccc(=S)n1O 59413,C(=O)(C#CC(C)(C)C)NCc1c(C(=O)NCC2(O)CCN(C)C2)nco1 59414,C(=O)(C(F)CC(C)(C)C)N1C(CNC(CC2(CSC)CC2)=O)C(C)CC1 59415,N1(C(C2=CC(C)(CC)C2)=O)CCOC2(CCS(=N)(=O)CC2)C1 59416,C1(C2(O)CCOC2)(C(N2CCC(F)(CNC(c3ncc[nH]c3=O)=O)CC2)=O)CC1 59417,n1(CC(=O)NCC2CC(NC(=O)C(O)C3CC3)C2)cc(Br)cn1 59418,c1(OC)cc(OC)[nH]c(=NCc2ccc(CN3CCOC(C(N)=O)C3)cc2)n1 59419,Cc1nc(C2CCCO2)sc1C(=O)N(C)CC1CCN(C(=O)CC2(O)CCC2)C1 59420,C1(C(NOC)=O)(OC(c2cccc(OC)c2)=O)CCN(N2CCCC2)CC1 59421,n1(CC2(C)CC2)nc(SC(F)F)nc1CCC1CSC1 59422,C1(NC(=O)NCc2nc(C(C)C)on2)CCCC(O)CC1 59423,C1(C(N2CC(CC(=O)OCC)C2)=O)C(C)OCCN1C(c1c[nH]c(=NC)o1)=O 59424,C1(N(C(c2c(C)ccc(F)c2)=O)CC)CCCN(C2CCc3ccc(Cl)cc32)C1C 59425,CC1(CCCO)CCCN1C(c1ccoc1CNC(c1cnn(C2CC2)c1)=O)=O 59426,C1(OCCNC(CC2C(C)CC2)=O)CCN(C(c2cnn(CCO)c2)=O)CC1 59427,C1(NC(c2sc(N(C)C)nc2C)c2n(CCCC)nnn2)CC(O)CC(C)(C)C1 59428,C(=O)(CC(C)(C)CNC(c1ccoc1Cl)=O)NC(c1nccs1)CC 59429,C1(c2ncc(C(=O)OC)s2)CCN(C(=O)N(C)C)CC1.C1CCS1 59430,C(=O)(C(C)C(C)COC)NCC#CC(=O)NCCC#C 59431,N1(C(=O)CCc2cscn2)CC(NC(C23CC(c4ccccc4)C2C3)=O)C(O)C1 59432,c1(C(=O)NCCC2(CNC(CC(COC)O)=O)CC2)cc(C)cc(Cl)n1 59433,C(CCCCC(=O)N1CCCC(CC(=O)NC(C)(C)CCCO)CC1)=CC 59434,C1(NC(C(CC)(C)OC)=O)CC=C(C(=O)NCC(C)(C)CO)C1 59435,N1(C(CCC=CC)=O)CCN(CC2(NC(=O)C(C)CC=CCC)CC2)CC1 59436,C1(C(=O)NCC(C)N(C(c2sc(C)c(Br)n2)=O)C)CNC(=O)C(C)(C)C1 59437,c1(C(=O)OC2(CC(=O)NC(c3ccnn3C)CC)CC2)cn(CCO)nn1 59438,N1(C(C(C)CC(C)(C)C)=O)CCC2CCN(C(c3cc[nH]c(=N)n3)=O)C2C1 59439,C1(NC(CCC(=C)C)=O)CCN(C(c2cccc(C(F)F)c2)=O)CC1C(C)C 59440,c1(-c2cn(C)nc2)cccc(NC(=O)NC2CCN(CC3CC3)C2)c1 59441,C(C)(CNC(=O)CC1CCOCC1)(C(C)C)NC(C(c1ccccc1F)C)=O 59442,c1(C(N2CCCC(C3CN(C(CS(=O)(=O)NC)=O)C3)C2)=O)ccc2ncnn2n1 59443,c1(NC(CC2CN(C(CC(C)=C(C)C)=O)CC23CC3)=O)cccc2occc12 59444,CC1(C)CCN(C(C23CC2COC32CCC2)=O)CC1CNC(=O)CC1CCOC1 59445,C1(C(C)C)(C(=O)NCCC2(O)CN(C(=O)Cn3cnnn3)C2)CCCO1 59446,c1(C(=O)OC)ncc(NC2(CNC(=O)CC(C)(O)c3ccccc3)CCCC2)nc1C 59447,C(=O)(C1=CCCN(C(=O)Cc2cc(C)cs2)C1)NCCCCC#CC 59448,Cc1[nH]c(C#N)cc1C(=O)NC1CCCCN(C(=O)CC2CC3CCC2CC3)C1 59449,CCCCC(C)C(=O)NCCOC1CN(C(=O)C(c2ccn(C)c2)C)C1 59450,CCCCC(C(=O)NCCN1CC(CF)C1)NC(C1CCOC(C)(C)C1)=O 59451,C12(NC(c3cnc(C4CC4)o3)=O)CCCC1N(C(c1ncccn1)=O)CCC2 59452,C1(C(=O)NC(c2nccs2)CC)CCCCC1(C)NC(=O)C=CC=C(C)C 59453,N1(C(C=C)=O)CC2CC(NC(=O)C(=Cc3ccccc3)CC)C2C1 59454,c1(CC(=O)NCCC(C)(C)NC(N)=O)ccnc(-c2nn[nH]n2)c1 59455,c1(CN2CCC(F)(C(=O)Nc3nc(OC)nc(O)c3)C2)ccc(C#N)cc1Cl 59456,Cc1ccc2c(c1)N(C(=O)C(CNC(=O)Cc1ccc(O)cn1)C(C)C)CC2 59457,CC(C)CCCC(=O)N1CCC(C=CC(=O)NC(CO)CC(C)C)CC1 59458,C1(C(=O)OC)CN(Cc2ccc(OC)c(Cl)c2)CCN1S(=O)(=O)CC(F)(F)F 59459,c1(OC)cc(Cl)ncc1C(N1CCN(C(c2oncc2C)=O)CC1CC#N)=O 59460,Cc1ncn(C)c1C(=O)N(C(C)CNC(c1cnn(CCO)c1)=O)C 59461,n1(C(C)(C)C)nccc1C(=O)NC1CCCC1NC(C1(N(C)C)CC1)=O 59462,C1(NC(c2cc(CO)[nH]n2)=O)CCN(C(c2ccccn2)=O)C12CCCC2 59463,C(C(C)CCCC(C)C)NC(C(CCC#C)NC(c1cn(CC)nn1)=O)=O 59464,c1(C(N2CCCCCC2CCO)=O)cnc2c(Br)cccn12 59465,N1(C(C=CC2N(C)CCC2)=O)CCC(NC(=O)Cc2ccoc2)C2(CCC2)C1 59466,C1(C(N(C)CC2C(C)OCC2)=O)C2CC3C(C2NC(=O)COC(F)(F)F)C13 59467,c1(OC)cc(NC(C2CCCC(NC(c3cnnc(O)c3)=O)CC2)=O)ccc1O 59468,C(=O)(C(CCC(C)C)OCC)N1CCC(C(N(CCC)CCOC)=O)(CC)CC1 59469,C(CN(C)C(C1CC1F)=O)(CO)(CO)NC(C(c1cccs1)SC)=O 59470,Cc1cc(C(=O)NC2CCC(C(=O)Nc3ncccc3C(F)F)C2)cc(F)c1 59471,Cc1nc(Cl)[nH]c(=NC2CN(C(c3ccc(N(C)C)cn3)=O)CC23CCC3)c1F 59472,C(=O)(C(=O)C(C)(C)C)NC1(CNC(c2n[nH]c(C)c2C)=O)CC1 59473,N1(C(c2c(C)noc2)=O)CCCN(CCCCNC(C2CC3CCC2O3)=O)CC1 59474,c1(C(=O)NC2CC(NC(c3sc(C)c(Br)c3)=O)C2)cccc(F)c1N 59475,CN=c1[nH]c(=NC2C=CC(CO)C2)[nH]c(=NC2COc3ccc(Cl)cc32)[nH]1 59476,N1(C(C2(COC)CC2)=O)CCCC(C(C)NC(=O)C(F)=C2CCC2)C1 59477,C1(N(C(=O)CC2(CO)CC2)CC)CCCN(C(=O)C=Cc2ccncc2)CC1 59478,N1(CC(=O)NC(C(=O)Nc2c(OC)nsc2)C)CCN(C)CC1 59479,c1(CC(CNC(COC2CN(C(C)=O)C2)=O)NC(c2cnc[nH]2)=O)ccccc1 59480,c1(NCCC(CCC)CCC)[nH]c(=NCc2sccc2C)nc2ncn(CC)c12 59481,c1(CCC(=O)NC(C)CCNC(=O)CCC2(C)N=N2)ccc2c(c1)NC(=O)CO2 59482,Cc1cc(C(=O)NC(CNC(c2c(C3CCC3)cnn2C)=O)CO)cc(F)c1 59483,C1(C(=O)NCCCNC(c2cnn3ccn(C)c32)=O)C2CCN(CC2)S1(=O)=O 59484,CCC(C)(C)C(O)C(=O)NCC1(OC)CN(C(=O)C(C)(F)c2ccccc2)C1 59485,C(C(F)(F)C(F)(F)F)CCC(=O)NCCOC1CCN(C(C(C)CO)=O)C1 59486,CC1(F)CC(C(=O)NCCS(=O)(=O)N2CCCC2C(N)=O)C1 59487,N1(C(c2nccc(COC)c2)=O)CC2(CCN(C(=O)C(C(C)C)NC=O)C2)C1 59488,C1(CC(=O)NC2C(CCC)CN(C(=O)COCP(C)(C)=O)C2)CC(C)(C)CCO1 59489,c1(C(N2CCC(N(C(CN(C)CC)=O)CCO)C2)=O)ccc(C(C)(C)C)cc1C 59490,N1(C(=O)C#CC2CCCCC2)CCC2C(CCCN2C(c2ccncc2O)=O)C1 59491,C(=O)(CCCOC1CC(NC(=O)CNC(C2CC2C)=O)C1)OC 59492,C(=O)(C(C)C(F)(F)C(F)F)N1C(CNC(c2cc(CC)cc(F)c2)=O)CCC1 59493,C1(C(N2C(CCNC(C(C)(C)CO)=O)CCC2)=O)Cc2ccc(Cl)cc2C(=O)O1 59494,c1(NC(c2nnnn2CC2CCOCC2)(COC(C)(C)C)C)ccc(Br)c(Cl)c1 59495,CC1(C(=O)NCC2(O)CC(NC(=O)CSC3CC3)C2)CCC(O)CC1 59496,Cn1cnc2c1CCN(C(=O)C(F)C(F)(F)F)C21CCN(C(=O)CC2(C)CC2)C1 59497,c1(C(N2CC(CN(C)C(C3CC3C(C)(F)F)=O)C2)=O)cc(C(N)=O)c[nH]1 59498,C1(C(=O)NC2(C)CC3(CCC4(C(C=C)C4)C(=O)N3)C2)CCOC2(CCCCC2)C1 59499,Cc1[nH]nc2cc(NC(=O)Cc3cccc4c3OCCC4)ccc12 59500,C12(C(=O)NCCNC(C(CC=CC)C)=O)CCC(C(=O)OC)(CO1)C2 59501,C1(C(=O)NCC2(C(F)F)CCN(C(Cc3c(C)ccs3)=O)C2)CCC2(CCC2)C1 59502,C1(N(C)C(C)C)CCN(C(=O)CC(=O)Nc2ncc(C(=O)OCC)s2)CC1 59503,c1(C(=O)NCC(C(C)C)NC(C(CC)(C)F)=O)cn2ccc(C)cc2n1 59504,c1(C(N2CCC(CN(C(CCC=CC)=O)C)C2)=O)csc(Br)c1C 59505,c1(C(=O)NC(C(C)NC(C(CC)(C)CC)=O)C)cccc(F)c1C#N 59506,C=CCCCC(C(=O)N(CCCC(=O)N(C)CCOC)C)NC(C)=O 59507,c1(COC)ccc(C(=O)NC2CCCC(C(N3CCSCC3)=O)C2)cc1 59508,C1(C)(C(=O)NC(CC)CC(=O)N(C2CCOC2=O)C)CC(=O)N(C)C1 59509,CN1CCC(C(=O)NCC2CC2NC(C2CC(NS(C)(=O)=O)C2)=O)C1=O 59510,C1(CC)CN(C(c2cc(Cl)ncc2F)C(=O)NC(C)(C)C)CC(=O)N1 59511,N1(C(c2ccc(C)o2)=O)CCC(CNC(c2nc(Cl)cs2)=O)C(O)C1 59512,CC1(C)CCCC(O)(CNC(=O)Cn2cc(C3(C)CCCO3)nn2)CC1 59513,C(=O)(C(CO)C(F)(F)F)N1C(C(=O)NCc2n(CCC)cnc2)CCOCC1 59514,C=CC(C)(C)CC(=O)NC1CC(F)(F)CC1NC(=O)Cc1cccc(F)c1F 59515,C1(CC(N2CCC(c3cnco3)CC2)=O)CNCCS1(=O)=O 59516,C1(C(=O)NCCN(CCC)C(c2cc(C(N)=O)n[nH]2)=O)CC12CC(C)(C)C2 59517,C(C(CNC(c1cncc(N)n1)=O)C(F)(F)F)NC(c1c(C)ccs1)=O 59518,c1(C(=O)NCCNC(c2ccc(C)cc2Cl)=O)cc(Br)cc2c1OCC2 59519,c1(CC(=O)NC(C2CCN(C(C3CCC3(C)C)=O)C2)C)coc2ccccc12 59520,Cc1nn(CCO)cc1C(=O)N(C)CC1CCCN1C(c1ccccn1)=O 59521,CCC(C)C(C)C(=O)N(C(C)CNC(=O)Cc1csc(C(=O)OC)c1)C 59522,CC1CN(C(C2CC2c2ccnn2C)=O)CC1NC(c1cnsn1)=O 59523,Cc1cc(C(=O)N(CCN(C(=O)C(N2C(C)CCC2C)C)C)C(C)C)cc(C)n1 59524,N1(C(CN(CCC)C)=O)CCC2(NC(C3CC3CF)=O)CCCC12 59525,CC1CN(C(=O)CCCCCN(C)C)CC(C)C1NC(=O)Cn1cccnc1=O 59526,O=C1NCC2(CCN(C(C3C=CCN(C(=O)C(O)CC(F)(F)F)C3)=O)C2)O1 59527,C1(C(=O)NC(COC(C)=O)CO)(COC)C=CCN1C(=O)C(n1ccnc1C)C 59528,CC1(C)CN(C(=O)CC(CNC(C2(C)CC3CC3C2)=O)C2CCC2)CCCO1 59529,C1(C(=O)NC2CC3CN(c4c(C)cncn4)CC32)CCc2ccc(F)cc2O1 59530,C1(C(=O)OCC)COCC1NC(=O)C(F)(F)Oc1ccccc1 59531,Cc1cc(S(N)(=O)=O)cc(-c2cc(N)c(C#N)cn2)c1C 59532,C(=O)(CCC(F)(F)F)N(C)CC1CCCN1C(C1CCS1(=O)=O)=O 59533,C12(C(N3CCCC(C)C3CNC(=O)Cn3cc[n+](C)c3)=O)CC=CCN1CCC2 59534,N1(CC(=O)NC(=O)NCC)CCCN(C(C2CCCC(OC)C2)=O)CC1 59535,Cn1nc([N+](=O)[O-])cc1C(=O)NC1(CCCNC(c2ccc(F)c(Cl)c2)=O)CC1 59536,c1(C(=O)NCCN(C(=O)CCc2ncc(C(C)(C)C)o2)CC)cc(SC)oc1C 59537,C(C)(CCC(=O)Nc1ccc(C(=O)NOCC=CCl)o1)OCC 59538,c1(NC(c2c(CCCN)ccs2)=O)nccc(CN2CCCC2)n1 59539,c1(C(=O)NC2CCCCCN(C(C(CC)(C)CO)=O)C2)cc(F)c(Cl)c(N)c1Cl 59540,CCC(C)CC(C)C(=O)N(C)CC1CCCN1C(c1ccccc1Cl)=O 59541,C1(NC(C(C(C)C)C#N)=O)CC2CCC1C(NC(C1(CCN(C)C)CC1)=O)C2 59542,C12(C(=O)NCCC(C)NC(C3(C#C)CCCC3)=O)CCC(C)(C(=O)O1)C2(C)C 59543,C1(CNC(CC2(C=C)CN(C(=O)Cc3cnn(C)c3)C2)=O)CC2(CCC2O)C1 59544,c1(C(=O)NCCCN(C(=O)CCC2CCCO2)C)ccc2c(Cl)nccc2c1 59545,C=CC(C)(C)C(=O)NCC1CCC(CN(C)C(C2CC2C(=O)OC)=O)CC1 59546,N1(C(CCCN(C(=O)CC#N)C)=O)Cc2cccc(O)c2C1 59547,c1(SCC)ccc(CC(N2CCOCC2CC(C(=O)C(C)C(F)F)=O)=O)cc1F.O 59548,C(=O)(CCCCC(F)(F)F)NCC(C(C)C)NC(CC(CC)C)=O 59549,c1(C(N2CCC(NC(CC(CC)O)=O)CC2C)=O)c(C)nn2cccnc12 59550,N1(C=O)CCC2CCC(C1)N2c1nnc(C2CCCC2)s1.c1(C2CCC2)cccnn1 59551,c1(CC)nc(C)c(NC(=O)CNC(C)(CNC(=O)OC(=O)C(C)(C)C)C(C)C)s1 59552,C1(C)(c2cn(CC3(C)CCC3)nn2)COCCN1C(=O)CC1CC(F)(F)CO1 59553,N1(C(c2ccon2)=O)CCC2(CCCN2C(c2ccn(CC(F)F)n2)=O)CC1 59554,N1(C(c2cc(OC)cc(F)c2)C(=O)NCC(F)F)CC2CCCCCC2(C#N)C1 59555,c1(C(N(C(CNC(c2cnsn2)=O)C2CC2)C)=O)ccc(=O)n2c1COCC2 59556,C(CCS(C)(=O)=O)(C(=O)N=S1(=O)CCCCCC1F)OC 59557,Cc1c(C(=O)NC2CCC(CNC(c3n[nH]cc3C(C)C)=O)C2)sc2nccn12 59558,Cc1cn2cc(CC(N3CCC(C)(CNC(=O)C(C)C)C3)=O)nc2s1 59559,C(N=c1[nH]nc(O)s1)C1CCCN(C(c2c(C)nn(CCO)c2)=O)C1 59560,N1(C(c2c(CCC)nns2)=O)CCCC(C)C1CCNC(c1ccnc(S)c1)=O 59561,N1(C(C(N)c2ccco2)=O)CC2COCC2(C(N2CC(O)C(F)C2)=O)C1 59562,C(CCN=C(NCC(c1ccccn1)(C)C)NC1CCCSC1)SC 59563,N1(C(C(CC2CCC2)NC(COC(CC)(C)C)=O)=O)CCCN(C2CC2)CC1 59564,c1(CC)cc(C(=O)NCC(CO)NC(C2(CSC)CCOCC2)=O)ncn1 59565,c1(C(N2CCCC(O)(CNC(C3C=CC=CC=C3)=O)C2)=O)ccc2nncn2c1 59566,C1(N(C)C(c2cn(C)nc2O)=O)CC2CCC(C1)N2C(=O)C(N)=O 59567,N1(CC(c2cccc(NC(=O)NC(C)=O)c2)=O)CC2CCC(CC2)C1 59568,C1(CC(=O)NCC2N(C(C(c3cnn(C)c3)C)=O)CC2)CC2(CC2)CO1 59569,c1(C(N(C(Cn2c(C)ncc2)C)C=O)C)cccc(Cl)n1 59570,C1(COCCO)(NCC2CCOCO2)CCCSC1 59571,c1(C(=O)NCC2(CNC(c3cnc(C4CC4)o3)=O)CC2)occ2c1CCCC2 59572,N1(C(C2CC(=O)NCC2)=O)CC2(NC(C3CCC3)=O)CCCC2(F)C1 59573,N1(C(CN(C)C(c2cccc(F)c2)=O)=O)CCCN(C(C2CC2(C)C)=O)C(C)C1 59574,Cc1nc2ncnn2cc1C(=O)N(CC(O)CN(C(=O)CO)C)C 59575,c1(OC)cc(OC)c(NC(C2CC(F)CN2C(c2cccc(O)c2)=O)=O)cc1Cl 59576,c1(CC(=O)NCC(CNC(c2cccc[n+]2[O-])=O)OC)nnc(S)n1C 59577,c1(C(N2CCCC(CNC(c3cccc(C)c3I)=O)C2)=O)cnc2snnc2c1 59578,c1(C(N2CC(F)CC(NC(C3CCCC(C)(C)O3)=O)C2)=O)ccc2nnnn2c1 59579,N1(C(C(C)(C)OC)=O)CCC(C)(CCNC(C2CC2C2CC2)=O)C1 59580,C(=O)(CCCCCc1ccccc1)NC1C(CNC(c2ccc(SC)s2)=O)C1 59581,CC1CC(=O)NC1C(N1CC(OCCNC(c2conc2C2CC2)=O)C1)=O 59582,c1(C(CNC(N2CC(CS(N)(=O)=O)C2)=O)F)ccc(Br)cc1 59583,c1(N2CCC3(C(C(=O)Nc4cc(N(C)C)cc(F)c4)C3)C2)ncnc2occc12 59584,Cc1nc(C)n(CC(=O)NC(c2ccc(F)cc2)CNC(=O)C=CC(F)(F)F)n1 59585,c1(N(C(C2C(C(=O)OC)C2)=O)CC#N)ccccc1NCc1cccc(Cl)c1 59586,c1(C(N2CCCC2CN2CCC(C(=O)NC)C2)C(=O)NC)cc2ccccn2n1 59587,c1(CC)cc(C(=O)NCCCCC(C)NC(=O)CCCc2ccccn2)ccn1 59588,N1(C(C(CNC(CC(CC)(C)C)=O)O)=O)CCN2CC(C)CC2C1 59589,N1(C(C2C(C)(Br)C2)=O)CCC(NC(c2nccs2)=O)C(F)C1 59590,CCCCC(C(=O)N1CC(C)C1C(=O)NOCCOCCOC)N(C)C 59591,c1(C(N2CCC(C(C)OC)CC2)C(=O)NCC(=C)C)cc(-c2cccs2)oc1C 59592,CC1=NOC(C(c2nnnn2CCCOc2ccccc2)(C)NC)C1.C1(CO)CC1 59593,C(=O)(CCCN=[N+]=[N-])N1CC(C)(OCC(=O)NC2CCC(CC(=O)OC)C2)C1 59594,Cc1ccc(C)c(C(N2CC(O)CCC2C(=O)NCCCN(C)C)=O)n1 59595,c1(C(N)=O)ccc(N2CCC(NC(c3nccc(Cl)c3O)=O)CC2)c([N+](=O)[O-])c1 59596,C(=O)(CCCCC1CC1)N(C1CCN(C(=O)CC2C(=O)NN=C2C)CC1)CC 59597,C1(C(=O)NCC(C)N(C)C(C2CCCN2c2cnccn2)=O)CCCC12CC2 59598,c1(C(N2CCC(OC)(CNC(=O)C(C)c3ccco3)C2)=O)ccc(F)c(F)c1N 59599,C(=O)(C#CC1CCCC1)NC(CC)CNC(=O)C(C1CCOCC1)OC 59600,c1(OCC)ccc(CC(=O)NC2CC(F)(CNC(=O)CC3CS(=O)(=O)C3)C2)cc1 59601,CC1(C)CCCC(C(=O)NC2CCN(CCCNC(=O)Cc3ccon3)C2)C1 59602,c1(CC(=O)NC2C(NC(c3c(CC)con3)=O)CC2)ccc(C)cc1F 59603,C(=O)(C1OCCn2ccnc21)NCC(CNC(c1c(NC)ccc(F)c1)=O)CO 59604,C=C(Cl)CN=C(NCC1(C)CCCCCCC1)NC(C1CC1)C1CC1 59605,CC1ON=C(C(=O)N2CCN(C(=O)CS(=O)(=O)N(C)C)CC2CO)C1C 59606,CCCCCCc1ccc(C(=O)NCC2CCN(C(C3CCS3(=O)=O)=O)C2)s1 59607,CC1CN(C)CCC1ONC(C1CCN(C(=O)CC2CCCCO2)CC1)=O 59608,CCC(CC(=O)N1C2CCC1CC(CNC(C1CCOC1)=O)C2)C(C)C 59609,N1(CC)N=C(C(=O)NCC2CC(O)(CNC(=O)Cn3nccc3C)C2)CCC1=O 59610,Cc1ccc(C(=O)N(CC(C)C(=O)N2CCC(CC(F)F)C2)C)n1C 59611,N1(C(C(C(C)C)SCC)=O)CC(CO)C2(C1)CN(C(c1cccc(=O)n1O)=O)C2 59612,c1(OC)c(F)ccc(NC(=O)C(C)N(S(C)(=O)=O)C)c1F 59613,Cc1ccc(O)cc1C(=O)NCc1nocc1C(=O)Nc1ccc(O)c(Cl)c1 59614,Cc1nc2cccc(C(=O)Nc3[nH]nnc3C3CCN(C(=O)OC(C)(C)C)C3)c2s1 59615,C1(NC(C(c2ccn(C)n2)C)=O)CC=C(C(=O)Nn2cncn2)C1 59616,c1(CNC(COCC(=C)C)=O)occc1C(=O)NC1CC=CCC1 59617,C(=O)(C1OCCc2ccccc21)NC(c1cn(CCOC)nn1)(C)C 59618,C1(CNC(c2c(NC)cccc2)=O)CN(C(c2ccc([N+](=O)[O-])o2)=O)CC1(C)C 59619,CCCC(C(=O)NCc1cccc(CNC(C2(C)C=CCC2)=O)c1)OCC 59620,c1(CC(C)C)ccc(C(N2CCCC2CN(C)C(C2CNC(=O)N2)=O)=O)s1 59621,Cc1cc(Cl)ccc1OC(CNC(C(C)OC(F)F)=O)CNC(=O)C(C)(C)C 59622,C(C)(C(CC(=O)NCC12CC(CN1C)C2)NC(=O)C(C)SC(C)C)OC 59623,C1(C)(C(N(CCOC)CCF)=O)C=CCN1C(C1CCOCC1OC)=O 59624,N1(C(CN2CC(CC)C2)=O)CCCC2(CCN(C(c3cc(C(F)F)cs3)=O)C2)C1 59625,c1(OC)ncc(NC(c2ccc(OC)c(C3CC3)c2)=O)c(C)n1 59626,c1(CNC(=O)CC2CC(NC3CCC(O)(C(=O)O)CC3)C2)cc2ccccc2o1 59627,C1(CNC(c2c(CC)con2)=O)(COC)CCN(C(C2CC(C)CO2)=O)CC1 59628,CCCC(F)(F)C(=O)N(CC(CC)NC(=O)C(O)CN(C)C)CC 59629,c1(CC)cnccc1NC(=O)NC(CO)C(C)NC(=O)COc1ccc(C)cc1 59630,C(CCC(=O)NCC(CO)NC(c1cnc(C2OCCO2)s1)=O)NC(N)=O 59631,CC1CC(C(=O)NCC2(C)CCOCC2)CN(C(=O)COCCCN(C)C)C1 59632,C(=O)(C1=CC2C=CC(C1)C2)NCCC(C)NC(c1c(OC)c(C)sc1)=O 59633,N1(C(c2n(C)c(C#N)cc2)=O)CCCC2(C1)CN(C(=O)CSc1n[nH]c(O)n1)C2 59634,CCCC(C)CC(=O)N(C(C)C(=O)NOCC1CCC1)C 59635,c1(N2C(CN(C(C(C)O)=O)C)CCC2)cc(C(F)(F)F)nc2ncnn12 59636,C=CC1CN(C(C2CN(C(c3cnn(C)c3Cl)=O)CC2OC)=O)CCO1 59637,C(C)(C(C)COC)(c1nnnn1CC1CCOCC1)NCC(=O)NC 59638,c1(C(N2CCOCC2CC2CC2)C(=O)NC(CC)C)ccc(N(C)C)nc1 59639,c1(C(=O)NCCN(C(=O)C(O)c2cnc[nH]2)CCC)ccc(Cl)c2cccnc12 59640,C=CC(C)CC(=O)N1CC(CO)(NC(=O)CSCc2c(C)noc2C)C1 59641,N1(CC(=O)NCC2CCN(C(c3cn(CCC)nn3)=O)C2)CCN(C)CC1 59642,c1(OC(C)C)ccc(C(=O)NC2(C)CN(C(=O)CC3CC(C(F)F)C3)C2)cn1 59643,C=CCC(C(=O)NCC(C)CNC(C1(CC=C)CCOCC1)=O)c1ccccc1 59644,c1(C(=O)NC2CC(F)(CNC(C(C)(C)OCC)=O)C2)cc(C)c(CC)o1 59645,c1(C(=O)NC2CCCC(NC(C(C)OCC=C)=O)C2)nc(C)ccc1O 59646,c1(C(=O)NC2CC3CN(C(C4CC(CC)(CC)C4)=O)CC32)cccc2c1COC2 59647,Nc1ccc(C(=O)NC2CCCC2NC(c2ncoc2C(F)(F)F)=O)cc1Cl 59648,N1(C(c2cccc(C(C)C)c2)=O)CC2(CC(NC(C3(C)CCC(=O)N3)=O)CO2)C1 59649,c1(C(=O)NC2CC(CC)(CC)N(C(=O)C3=NOC(C)C3)C2)c(C)ccc(C)c1O 59650,N1(C(C2N(C(c3ccc(C(C)=O)[nH]3)=O)CC=CC2)=O)CCOC(C)(C)CC1 59651,c1(C(N2C(CNC(CCc3c(C)noc3Cl)=O)CC2)=O)cnc2c(c1)OCCN2 59652,Cc1cnc(C(C)NC(=O)C(COC(C)C)NC(=O)CC(=O)NC2CC2)o1 59653,C1(NC(CCNC(C)=O)=O)C2CC3CN(C(=O)COC(CC)CC)C1C3C2 59654,N1(C(C(CCC)N(C)C)=O)CCC2(C1)CN(C(C1CC1(C)C)=O)C2 59655,N1(C(CCC2(C)CN(C(CNC(C3C(C)C3)=O)=O)C2)=O)CC2CC(O)CC1C2 59656,C1(C(N2C(C(=O)NC)CC(O)C2)=O)CN(C(=O)CC2C=CCCC2)CCC1(C)C 59657,O=C1NCc2c1ccnc2C(N1CC(CNC(C2CC(O)C2)=O)C(O)C1)=O 59658,C1(C(N2C(C)(C(=O)NCCC3CCN(C)C3)C=CC2)=O)CCCC(C#N)C1 59659,C(C(C)(C)CC(=O)NC1CN(C)CC1C)NC(C1(CC)CCC1)=O 59660,c1(C2(NC(=O)NC(C3CCCC3C)C)CCC2)cccc(Br)c1 59661,Cc1cccc(NC(C2CCN(C(=O)Cc3cc(F)ccc3Br)C2)=O)c1[N+](=O)[O-] 59662,C1(C)(CNC(=O)OC(C)(C)C)CCC(NC(=O)C(=O)NCCN2CCCC2=O)C1 59663,N1(C(c2cncc(C#C)c2)=O)CCC(NC(=O)C#CC2CC2)C12CCC2 59664,N1(C(c2cccc(O)c2)=O)CC2CCN(OC(c3cccc(CC)n3)=O)CC2C1 59665,c1(CC(=O)N(CC(CN(CCCCCC=C)C)O)C)nc2ncccn2n1 59666,C1(C(=O)NCC(=O)OCC#C)(NC(C2CC2(Cl)Cl)=O)CSC1 59667,c1(NC)cccc(C(N2CCC(CN(C)C(C3CC(C)(F)C3)=O)C2)=O)n1 59668,Cc1sc2ncc(C(=O)NC3CC3CNC(c3ncoc3C(C)(C)C)=O)n2c1C 59669,Cc1cc(C(=O)NCC2C3CN(C(c4cc(Cl)c[nH]4)=O)CC23)cc2nc[nH]c12 59670,c1(COCC(=O)NCC(CNC(CCNS(CC)(=O)=O)=O)O)ncc(C)o1 59671,n1(C(C)C)cc(C(=O)NCCC2CCN(C(=O)CCN3CCC3)C2)c(Br)n1 59672,C=CCC(C)(C)CC(=O)NCc1cncc(C(=O)NC2CN(C(N)=O)C2)c1 59673,C1(CC(=O)NC(CC(=O)NCCC(C)(C)O)C2CC2)CC2(CC2)CO1 59674,Cc1ccc(F)c(O)c1C(N1CCC2C(NC(c3c(Cl)cnn3C)=O)C2CC1)=O 59675,C1(C(N2CCOC(CC)C2)=O)(CNC(C(COCC)C)=O)CC12CCC2 59676,c1(C(N2CCN(CC(=O)NCC3N(CC)CCC3)CC2)=O)cc(F)cnc1O 59677,c1(CC(=O)NCC2(C(C)OC)CC2)cn(C)nn1.C(=O)C1CC1 59678,CCCCC(=O)NC(C)C(c1ccccc1)NC(C1CC(=O)C1C)=O 59679,c1(C(=O)NCCC(C)NC(c2ccc(CO)o2)=O)ccc(OCC(F)(F)F)cc1 59680,c1(OC)cccc2sc(C(=O)NCC(O)CNC(=O)C(C)n3cccn3)cc12 59681,c1(C(=O)NC2C(NC(C3C(C)C3)=O)CCC2)cnn(C)c1Cl 59682,C1(N(C(CC(=C)I)=O)C)CCC(n2cc(-c3ccc(OC)s3)nn2)CC1 59683,C(=O)(N=c1nc2cccc(OC)n2[nH]1)C1CC(=C)CN1C(c1cc(C)n(C)n1)=O 59684,C1(NC(C2(C)CC(=C)C2)=O)C=CCC(C(=O)NCCc2ccn(C)n2)C1 59685,c1(OC)cc([N+](=O)[O-])ccc1C(=O)NC1C2CC1CN(C(=O)C(C)C1CC1)C2 59686,C1(NC(COCCC#C)=O)(CO)CCN(C(=O)CCC2CCCCN2C)C1 59687,c1(C(=O)NC2C(CNC(=O)CC3CCOC3)C2)c[nH]c2cc(Cl)ccc12 59688,CC1CC(CNC(C2CC3CC3C2)=O)CCN1C(=O)CCOC1CCOCC1 59689,C1(C)(C(=O)NCC(CC(C)C)NC(CCC(=C)Cl)=O)CCCC1(F)F 59690,c1(C(=O)NC(C(CCc2ccccc2)NC(CC=C=C)=O)C)cnc2sccn12 59691,c1(OC)cc(C(=O)Nc2cc(C)cc(C)c2Br)c(N)cc1Cl 59692,c1(C(N(CC(C)C(N2C3CCC2CC3)=O)C)=O)cccc(F)c1N 59693,C(CC(=O)N1CC(C)(C)C12CCC2)(CC(C)C)NC(CC(COC)(C)O)=O 59694,C1(C(=O)NCCCN(C)C(c2ccc(Cl)c(O)c2)=O)COc2ccccc2C1 59695,N1(C(C2CC(=O)CN2C(=O)CC2CCC=CCC2)=O)CC2(CCNC2=O)C1 59696,c1(C(=O)NCCCCNC(C(C2CCCOC2)OCC)=O)cnn(CCO)c1 59697,C=CC(C)CC(=O)NC(C1CN(C(=O)CCc2cncnc2)C1)C 59698,C1(NC(=O)NCC2(CCO)CN(C(=O)OC(C)(C)C)C2)CCc2ccnn2C1 59699,c1(C(N2C3CC(NC(CN4CCC(C)C4)=O)(C3)C2)=O)cccc2c1OCC2 59700,N1(Cc2c(F)cc(C#N)cc2Br)CCC(N)c2cc(Cl)ccc21 59701,c1(C(N2CC3C(N(C(=O)CC4(C)CC4(Cl)Cl)C)C3C2)=O)cncn(C)c1=O 59702,c1(C(=O)NCCCN(C(CSCC#C)=O)C(C)C)ccc(Cl)c(OC)c1 59703,Cc1ccc(C(=O)NC2CC2C(=O)N(CCO)C2CC2)cc1[N+](=O)[O-] 59704,c1(C(N2CCC(NC(CCCN(C)C)=O)C2C(C)(C)C)=O)nccc2cc[nH]c12 59705,C(CC(=O)NCc1cc(C(N)=O)no1)(C(F)F)NC(CNC(C1C(C)C1)=O)=O 59706,N1(C(CCC2(C)CCCN2C(=O)C(O)C2CC2)=O)CCCCCCCC1 59707,Cc1nc2ccc(C(N3CCCC3c3cn(Cc4cccc(Cl)c4)nn3)=O)cc2o1 59708,Cc1n[nH]c(C)c1CC(C)C(=O)NC(C)CC(C)NC(=O)C(C)O 59709,C(=O)(C(CNC(=O)CC(C)(F)F)CC1CC1)NCc1ccc(CC)o1 59710,C1(CCNC(c2ccc(C(F)F)s2)=O)CCCCN1C(C12CCC1C2)=O 59711,c1(C(N(CCNC(c2cc(C)oc2)=O)CCOCCO)=O)c[nH]ccc1=O 59712,CCCC(F)C(=O)NC1(CCCNC(=O)CCCNC(=O)OC)CC1 59713,CC(C)(C)C(=O)C(=O)N1CCN(C(c2sccc2F)=O)CC1CC1CC1 59714,CON1CCC(CC(=O)NC2CC(F)(CNC(C3CCN3S(C)(=O)=O)=O)C2)CC1 59715,C1(NC(c2nccc(OC)c2)=O)CCCC12CN(c1ccncn1)C2 59716,C1(CC=C)(NC(C2CC2c2ccccc2Cl)=O)CCN(C(=O)C(F)(F)COC)C1 59717,C1(C(=O)OC)CCCCCN1C(c1ccc(OC)nc1)C(=O)NCCCC1CC1 59718,C1(SC)CCC(N=c2[nH]c(N3CCCC(C)(C)CC3)nc3c(F)cccc23)C1 59719,CC(C)(C)C#CC(=O)N1CCN(C(=O)CC2CCS(=O)(=O)CC2)C(CF)C1 59720,C1(NC(c2nc(CC)oc2)=O)CN(C(c2ccccc2NC)=O)CC1NC(N)=O 59721,C(CCC(=O)NC(CN(C)C)C(=O)NCCCC1(O)CCC1)OCCOC 59722,Nc1ccc(C=CC(=O)NCC2CCCN(C(C3CCCOCC3)=O)C2)cc1N 59723,CCC(C)C(O)C(=O)NC1CC(CCNC(c2cc(C3CC3)ccc2Cl)=O)C1 59724,C(CC(C(C)(C)C)NC(=O)Cn1cnnc1)N(C(c1c(C)nccc1)=O)C 59725,CCC(CC)(CCNC(=O)C(C)Cn1ccnc1)NC(c1cc(F)n(C)n1)=O 59726,Cc1c(Cl)c(C(N2CCC(C)(NC(C3CC34CCCC4)=O)C2)=O)nn1C 59727,N1(C(C(=O)NC(C(=O)N(CC)CC)C)=O)CCCC2(C=CCO2)C1 59728,C12(C(=O)OC)CC1CN(C(c1ccc(N(C)C)nn1)C(=O)NCCC1CC1)C2 59729,C1(C(N2CC(O)(C(C)NC(=O)Cc3csc(C(C)C)n3)C2)=O)(COC)CC1(F)F 59730,CC(C)(C)CC(N)CCN1CCC(C)(C)C1=O 59731,N1(C(CCN(CCCCC)C(C)C)=O)CCCC1CNC(=O)C=C(C)C(F)F 59732,N1(C(Cc2n(C)nnc2)=O)CC2(C(=O)NC3CC(CO)C34CCC4)CCC1CC2 59733,c1(CNC(N(C2CCCOC2)CCC)=O)cnc(COC)s1 59734,c1(OC)nccc(C(N2CC=CCC2C(=O)NCC2C(C)C2(F)F)=O)n1 59735,C(=O)(C(F)(F)CCCNC(C)(C)C)NCC1(C)CCCN1Cc1ccccc1 59736,CC(C)CC(C(=O)N1CC2CC(NC(C3(C(C)C)CC3)=O)CC1C2)C(N)=O 59737,c1(SC)c(C(=O)N(c2cccn(C)c2=O)C)cccc1Br 59738,N1(C(C(CC(C)C)O)=O)CCC2(CC(NC(c3cc(C4CC4)ccc3F)=O)C2)C1 59739,C1(C(=O)NCCCNC(=O)CNC(C2CCOCC2)=O)CN=C2N=CNN2C1 59740,c1(C(=O)NCCCN(C)C(C2CC(C)(CN)C2)=O)ccc2c(c1)C=CS2(=O)=O 59741,C1(CNC(c2n(C(CC)C)ncc2)=O)CCCN(C(=O)C(C)(C)CC)C1 59742,C1(C)(C(=O)Nc2scc(C(=O)OC)n2)CCN(C(=O)CNC(=O)OC)CC1 59743,C(=O)(C(F)C(F)(F)C(F)(F)F)N1CC(CNC(=O)C2=NNC(=O)C2)CC(C)(C)C1 59744,C(C(N=c1[nH]c(Cl)ncc1[N+](=O)[O-])C1CC1)NC(C1N(C(CCC)=O)CCC1)=O 59745,n1(CC)cnc2c(NCc3cnc(C)o3)nc(N3CCOC(C)(C4CC4)C3)nc12 59746,C(C)(C)(C(=O)NCC1CCN(C(C2CCC2C)=O)C1)NC(=O)NCCC 59747,C1(Cl)(C(=O)NCC2(NC(c3nc(CC(C)C)sc3)=O)CCOC2)CC12CCC2 59748,c1(NC(C(CC)NC)c2nnnn2C)cc(CNC(=O)OC(C)(C)C)ncn1 59749,c1(C(=O)NCCC2(CNC(C(C)=C3CC3)=O)CC2)ccc2nc(S)oc2c1 59750,C(CNC(=O)CC1(N(C)C)CC1)(C(C)(C)C)NC(C(C=C)C)=O 59751,c1(C(C(=O)NCCCSCCO)N(CC(C(=O)OC)C)C)cc(C)c(C)c(Br)c1 59752,[N-]=[N+]=Nc1ccc(C(=O)NCC2CCCN2C(C2CCC3CCCCN23)=O)cc1 59753,C1(C(N(C2CC=CC2)C)=O)CC1C1CN(C(c2cc(Cl)cs2)=O)C1 59754,C1(CNC(c2n(C)ncc2)=O)CN(C(c2cc(F)n(C)n2)=O)CCN1C 59755,C1(CC(=O)NCC=C=C)CN(C(C2(O)CC(CF)C2)=O)CCO1 59756,c1(CC(=O)O)cn(C2(N3C(NC(c4ccc(-c5cccs5)[nH]4)=O)CC3)CC2)nn1 59757,N1(CCNC(c2c(CC)non2)=O)CCCN(C(C2CC(C#N)(OC)C2)=O)CC1 59758,C12(CNC(=O)NC(C3CS(=O)(=O)C3)C)CCC(C)(CO1)C2 59759,n1(CCOC)nc(OC(=O)C(c2cnn(C)c2)=O)c2c1CCOC2 59760,N1(C(c2c(CC)n[nH]c2)C(=O)Nc2ccccc2C)CCC(O)CC1(C)C 59761,O=C(CC(C(F)F)n1cccn1)NC1CCN(c2cc(C(N)=O)ncn2)C1 59762,C1(NC(C=CC(C)C)=O)(CNC(c2cc[nH]c2C2CCCC2)=O)CCOC1 59763,c1(C(=O)OCC)ccc(N2C(=O)N3CCC3C2)cc1.C1(NC)CCCCO1 59764,N1(C(c2c(CC)cns2)=O)CCN(C(=O)CCc2cncc(F)c2)CC1CCO 59765,C1(C)(COC)CC(NC(=O)CSc2nnnn2C)CN1C(c1cc(O)n(C)n1)=O 59766,C1(NC(C2(C)C=CCN2)=O)CCCC12CCCC2 59767,N1(C(C(CSCC)NC(c2ccsc2)=O)=O)CCC2(CCC(OC)C2)C1 59768,C1(c2cnc(C)[nH]2)NC(=S)N(C2CC2)C2=C1C(=O)NC(C)C2 59769,C1(C)(C(N(CCC)CCNC(=O)COCC2CCCOC2)=O)CCC(C)=C(C)C1 59770,C1(NC(c2cc(C)sc2C)=O)CC(NC(=O)C(=O)NCC(F)F)C12CCOCC2 59771,c1(C(NN)=O)ccnc(CNC(C2CC=CCC2NCC2OC3CCC2C3)=O)c1 59772,CCC(N=c1[nH]c(=NC(C)c2cnccc2C)[nH]c2ncn(C)c12)C(C)C 59773,N1(C(CCN(CCC)C)=O)C2CCC(C2)C1CC(=O)NC(c1cc[nH]n1)CC 59774,C#CCC(C)(C)C(=O)N1CC2(CC(CNC(c3cc(N)cnc3C)=O)C2)C1 59775,N1(C(Cc2c(OC)ccc(C)c2)=O)CC(C2CN(C(C3CC(C)CCO3)=O)C2)C1 59776,CC1CCN(C(c2cnn(C)n2)=O)C1CNC(=O)CCCN1CCCCC1 59777,C1(NC(CSC(C)(C)C)=O)CC(N=c2[nH]ncs2)C12CCOCC2 59778,C1(N(C(=O)CC2C=CCCC2)CC=C)(CCc2nn[nH]n2)C=Cc2[nH]ccc21 59779,Cc1ccc(OCC(=O)NC2CC3CCC2(NC(c2cncnc2)=O)C3)cc1C 59780,C=CC1CN(C(c2cccc(COC)n2)=O)CC1NC(C12CC(F)(C1)C2)=O 59781,N1(C(C(CCC)CNC(C2C3CCC(F)C23)=O)=O)CCC(O)C12CCC2 59782,C1(C(C)C)CCc2c(sc(NC(c3cc(C4CC4)ns3)=O)c2C#N)C1 59783,C(=O)(CCS(C)(=O)=O)NC(C)C(C)C(=O)NC1(C(N)=O)CC1 59784,c1(SCC)nccnc1C(=O)NC1C=CC(CNC(C2COC(=O)N2)=O)C1 59785,c1(-c2cc(C)nn2C)cccc2c1CCN(C(=O)CCOC1CCCCC1)C2 59786,C(=O)(CS(C)(=O)=O)N(CC(=O)NCC(COC)(C)O)CC(C)C 59787,c1(C(N(C(CCNC(c2c(C)noc2C2CC2)=O)C)C)=O)cn2c(n1)CCC2 59788,N1(C(C(C)O)=O)CC2CC(C)N(C(c3cc(N)ccc3Br)=O)C2C1 59789,CC(C)(CC(=O)N1CCN(C(c2ccc(N)c(F)n2)=O)CC1)C(F)F 59790,C1(C(=O)NCC2(CCC=C)CCOCC2)CCCN(C(C)C(C)(C)C)CC1 59791,c1(C(=O)NC2CN(C(c3c(C)n(C)cc3)=O)C(C)C2)c(F)cccc1Br 59792,C#CCCN=C(NCC(O)Cc1ccccc1)NCC1(C)CCCCO1 59793,c1(C(N(C)CC2CCN(C(c3c(C(C)C)csc3)=O)C2)=O)ncc(N(C)C)cn1 59794,c1(C(=O)NC2C(CNC(C(C)(C)N3CCCC3)=O)CCC2)cnc2n1CCCC2 59795,CC(C)C(O)C(=O)NC1CCC(NC(C2(Cc3ccccc3)CCC2)=O)C1 59796,c1(C(N(C2CCN(C(C3(SC)CC3)=O)C2)CC)=O)ccc(Cl)c(C(=O)NC)c1 59797,C(CC(F)F)(C(=O)NCC1(C)CC(C)(C)C1)NC(c1cn(C)nn1)=O 59798,C1(NC(=O)CCn2cnnn2)CC(F)(CNC(C2CCOC2)=O)C1 59799,c1(C(N2CCC3C(NC(CCCC(=C)C)=O)C32)=O)cc2c(C3CC3)cccc2[nH]1 59800,c1(C(=O)OC)cnc(OC2CN(C(=O)COC(C)(C)C(F)(F)F)CC2C)c(F)c1 59801,N1(C(C(COC)C)=O)CC2(C)CN(C(c3ccn(CC4CC4)c3C)=O)CC2(C)C1 59802,CCCCCC(O)C(=O)N1CCC(NC(=O)COc2ccc(C(C)C)c(C)c2)C1 59803,c1(C(=O)NCCCCc2cn(-c3ccc(Br)cc3Cl)nn2)ccc2ncsc2c1 59804,C12(C(=O)NCC3(NC(CCC=C=C)=O)CCCC3)CCCCC1C2(F)F 59805,Cn1cc2cccc(C(N3CCCC(NC(c4cnc(C5CC5)s4)=O)C3)=O)c2n1 59806,N1(C(c2cc(N)cc(F)c2)=O)CCCC2CN(Cc3ccc(F)cn3)CCC12 59807,n1(CC(=O)N(C(C)C2CC2)C2CC2)nc2ccccn2c1=O 59808,C=CCC(C)(C)CC(C(=O)NC1(C)CC1)N1CCC(C)(F)C1 59809,Cn1ncc2nc(O)c(C(N3CC(CNC(=O)Cc4cccs4)C3)=O)cc12 59810,C1(CC)CN(C(C2CC(C#N)(OC)C2)=O)CCN1C(=O)CCc1cccc(C)n1 59811,Cc1cc(CC(=O)NCCCN(C(=O)C(C2CC(C(F)F)C2)C)C2CC2)n(C)n1 59812,C(CNC(C1CCCN1C1CC1)=O)(CC(F)(F)F)NC(CN(CC(C)(C)C)C)=O 59813,c1(C(=O)NC2CCCN(C(C3CCCCC3)=O)C2)c(O)cc(Br)cc1F 59814,N1(C(C2C3(CC(OCC)C3)C2)=O)CCC(NC(=O)C=C(Cl)Cl)C2(CCC2)C1 59815,C(=O)(C(C)C(CC)CC)NCC(CC)NC(=O)CCCC1CCOCC1 59816,c1(CCC)cc(C(=O)NC(CNC(=O)C(C)CN2CCCCC2)CC)n(C)n1 59817,CC(O)C(C)C(=O)NCCOC1CN(C(c2nccnc2-n2ccnc2)=O)C1 59818,CCC(C)C(C(=O)NC1(CO)CC2CCCC12)NC(=O)C=CC(F)(F)F 59819,c1(C(C)=O)ccc(=NCCNC(c2ccc(-c3cccs3)cc2)=O)[nH]c1 59820,Cc1cnc2c(cnn2CC(=O)NCC2CCC(NC(=O)CC#N)C2)c1 59821,C12(NC(CCCOC)=O)CCC1CN(C(=O)CCN1CCCS1(=O)=O)C2 59822,N#CC1CN(Cc2ccccc2)CC1NC(=O)NCCc1ccccc1Br 59823,C(=O)(C1=C(Cl)CCCC1)N1CCCC(C)(C(=O)NC(c2nc(C)on2)C)C1 59824,C1(N(C(C(CC#C)C)=O)C)CCCCN(C(c2onc(CC)c2C)=O)C1 59825,C1(CC(=O)NC2CN(C(C(C=CC)O)=O)CC(C)C2)C2CC3CC(C2)CC1C3 59826,CN1CCC(O)C(c2nnc(N3CCN4CCC3C4)n2CCC#N)C1 59827,N1(C(c2c(C)nc(COC)s2)=O)CC2CCN(C(=O)CCC3CC3(Cl)Cl)C2C1 59828,CC1(C)CC(C)(C(=O)NCC2CCCCC2NC(C2CCCS2)=O)C1 59829,CC1(C(N2CC(N=[N+]=[N-])C2)=O)CCN(C(C2CCCO2)=O)CC1 59830,Cc1ccc(C(=O)N(C2(C(=O)N(CCCC3CCCO3)C)CC2)C)c(F)c1 59831,C(=O)(C1=NNC(=O)CC1)N1CCCC(NC(C2CCCC(C(=O)OC)C2)=O)CC1 59832,c1(C(N2C3C(N(C(C=C(C)C)=O)C)CC(C3)C2)=O)cc([N+](=O)[O-])cn1C 59833,c1(CCC(=O)NC(C)CNC(=O)C2CC2)ccc(Br)cc1 59834,Cc1ccc(-c2ccc(CNC(c3cccn4c(O)nnc34)=O)nc2)c2cn[nH]c12 59835,CCCCCCCC(F)C(=O)NCC1CCN(C(C2(C)CCCC2)=O)C1 59836,N1(C(CNC(C(C)n2cnnn2)=O)=O)CCN(C(=O)CC2CCCC23CC3)CC1 59837,N1(C(C2CC3(CC(C)C3)C2)=O)CCN(C(c2cnc(C3CC3)[nH]2)=O)C2COCC12 59838,C1(CCOC)CCN(C(=O)Cn2c([N+](=O)[O-])cnc2C)CC1(F)F 59839,N1(CCCC(CC)=O)CCN(Cc2ccncc2)C2CC12 59840,N1(C(C2N(C)CCC2)=O)CC2CC1C2NC(=O)CC1CCN(CC(F)(F)F)C1 59841,c1(C(N2CC(OC)(CNC(C3(CCF)CC3)=O)C2)=O)ccnc(F)c1 59842,C1(NC(C2(C)CCN2C(C2(F)CC2)=O)=O)CCCC(O)C1 59843,C1(CN(C)C(C2CC2F)=O)CN(C(=O)CCOC2CC2)CC12CC2 59844,c1(C(=O)NCC(CC=C)NC(=O)Cc2cncnc2)cccc2ncc(C)cc12 59845,C1(NC(c2cc(C#N)ccc2C)=O)CCCC12CN(C(C1C(C(=O)OC)C1)=O)C2 59846,N1(C(C(C)N(C)C)=O)CCCC(C)(CNC(=O)CCN(C)Cc2ccccc2)C1 59847,C1(C)(CNC(C2N(C(Cn3ncc(CC)c3)=O)CC=CC2)=O)CC2CCC1C2 59848,N1(C(CSCCC)=O)CC(NC(C23CCC(F)(CC2)C3)=O)C2CCCCC12 59849,c1(C(C)C(=O)NC(C)(C)CNC(=O)Cc2nccn2C)ccc(Cl)cc1 59850,C(=O)(C#CC(C)(C)C)N(C(C)CNC(c1snnc1C1CC1)=O)CC 59851,Cc1ccc(Cl)cc1C(=O)NCCC1(O)CN(C(C2COCC(C)O2)=O)C1 59852,N1(C(C(CSC)OC)=O)CCCCCC(NC(c2cncc(OC(C)C)c2)=O)C1 59853,S(=O)(=O)(c1cnc(NCC(c2nccs2)C)c(Cl)c1)N1CCn2c(C)ncc2C1 59854,CCC(C)C(O)C(=O)N1C2CCC1(CNC(C1(C)CCC1)=O)CC2 59855,c1(C(N2CCN(C(C(C)=CC)=O)C3C2C3)=O)cccc2c1CCOC2 59856,C1(CNC(CC2C(C)C2)=O)(CO)CCN(C(c2ccc([N+](=O)[O-])o2)=O)CC1 59857,C(CNC(=O)Cc1cnnn1C)(CC(F)(F)F)NC(C(C)SC)=O 59858,C12CCCCN(C1)C(=O)CC2.C1(NC2(c3ccn(C)n3)CC2)CCCC12CCC2 59859,c1(NC(CC2CC(NC(c3n(C=C)nnc3)=O)C2(C)C)=O)ccc(F)cc1O 59860,Cc1nc2cc(C(=O)NC3(CNC(=O)CC4COC5CC4C5)CC3)[nH]c2s1 59861,c1(SCC)nc(N2CC(Nc3ncc(C)cn3)C(O)C2)ncc1F 59862,N1(C(C(C)OCC#C)=O)CCN(C(c2c(C)noc2C)=O)CC1c1ccccc1 59863,N1(CC)CC(NC(=O)C(CC2CCCC2)NC(=O)C(C2CCOCC2)=O)C(C)C1 59864,N1(C(C2(C(=O)OC)CCCC2)=O)CCCC(C)(NC(C2CC(OC)C2)=O)C1 59865,CCC(C)C(O)CC(=O)NC1(CNC(c2n[nH]c3ccccc23)=O)CC1 59866,N1(C(C=C(C)C(C)C)=O)CC2C(CNC(C3CC4CCC3O4)=O)C2C1 59867,N1(C(C2(C#C)CN(C(=O)CN3C(=O)CCCC3=O)C2)=O)CC2(CC2)CC1CO 59868,C(=O)(CS(=O)(=O)C1CC1)NCC(C(C)C)NC(C1(CC(=O)OC)CCCC1)=O 59869,C(=O)(C(CCC(C)(C)C)N(c1ccccc1C(C)C)C)NC1CC(C(=O)OC)C1 59870,C(c1ccccc1Cl)=CC(=O)NC1CCCN(C(=O)CC2COCCO2)CC1 59871,C(c1ccncn1)=CC(=O)NC(C(C)NC(c1cscc1F)=O)C 59872,C1(CC(=O)N(C2CC(NC(c3cc4ccsc4s3)=O)C2)C)CC(C)(C)OC1=O 59873,C1(CC)CC1N=c1[nH]c(N(C)Cc2nn(C)c3ccccc23)nc2ccsc12 59874,c1(C2(C(=O)NC(CC)C(C)(C)O)CC2)ccc(C)c(Cl)c1 59875,c1(N2CCC(C)(C)CC2)ccncc1S(=O)(=O)N1CC(C)(C)OCC1CO 59876,c1(C(=O)NC2CC(NC(C(C=C=C)C)=O)CC2O)cc(O)nc(C)n1 59877,c1(C(N2CC(O)(CCNC(C3(COC)C=CCC3)=O)C2)=O)[nH]c(O)nc1C 59878,CCCC(C(=O)N1CCOC(CCNC(=O)C(F)=C(C)C)C1)N(C)C 59879,N1(C(CCNC(=O)OC)=O)CCC(NC(=O)CC2COCCN2C)C1C(C)(C)C 59880,C1(C(=O)NCCC(C)CCO)(OC)CCN(C(C2(OC)CCCCC2)=O)C1 59881,c1(-n2cc(C3(NC(=O)C(c4cccnc4)O)CCC3)nn2)ccc(Cl)cn1 59882,N#Cc1cc(C(N2CCC(CC(=O)Nc3ccc(F)c(F)c3Cl)C2)=O)ccc1F 59883,C1(NC(CCN(C(c2c(C)csc2)=O)C)=O)CCOC12CCOC2 59884,N1(C(=O)NC(c2ccncc2Br)C)CCC2CCC12c1cccs1 59885,N1(C(Cc2c(C)cco2)=O)CCCC(CCNC(c2ccc(F)cc2)=O)CC1 59886,C1(C)(C(=O)NCC(C(=O)OC)(C)C)CCCN(Cc2cccc(O)n2)C1 59887,CC(C)CC(C)N(C(=O)CONC(c1coc(C(F)F)c1)=O)C 59888,C(=O)(C(F)C(C)CNC(c1cc(C)c(N)cn1)=O)N1CCC(C(=O)OCC)C1 59889,C(=O)(CC1C(=O)Nc2ccccc21)N1CC(C)C(NC(C2CSCC(=O)N2)=O)C1 59890,C(CCN=C(NCC1(C#N)CC1)NC1CCNC(=O)C1)OCC 59891,C(=O)(C1CNc2ccccc21)NCC1C(C)(C)CCN(C(C23CC(CO2)C3)=O)C1 59892,C12(NC(C3CCCCN3C(C3CCC3)=O)=O)CC(C1)N(C(=O)CCCCO)C2 59893,c1(C(=O)NC(C2CC(NC(C3(Cl)CC3(C)C)=O)C2)C)cc(-c2cnn(C)c2)[nH]n1 59894,CC1CN(C(=O)C(=O)C2CCCC2)CC(C)CN1C(c1cc(C(N)=O)co1)=O 59895,c1(C(=O)Nc2ncc(CO)cc2Br)cc(Cl)cc(Cl)c1F 59896,Cn1cc(C(=O)NCC2CCCC2NC(c2ccccc2Cl)=O)nc1O 59897,c1(C(=O)NC(CN(C(=O)C(CC)OC)CC)C)ccnn1C(C)(C)C 59898,C1(C(N2CCCCC2C2CC2)=O)C2CC(O)C(C2)N1C(=O)C(O)CC(F)(F)F 59899,CC1=NN(C)C(=O)C1CC(N1CCC(NC(c2ccnn2C(C)C)=O)C1)=O 59900,C1(O)(C(=O)NCC(N(C(c2ncn(CC)n2)=O)C)C2CC2)CCC(C)CC1 59901,c1(OCCCN(CC(O)CN(C)C(=O)C2CC2)C(C)C)ccc(F)cc1Cl 59902,c1(C(=O)NC(C(C)NC(=O)CCN2CCCC2)C)coc(C(N)=O)c1 59903,N1(CC(=O)NCC(C)NC(c2c(CC)c(C)sc2)=O)CCCCCCC1=O 59904,C(=O)(CC(C(F)(F)F)NC(=O)COCC=C)NC1(CC#C)CC1 59905,N1(C(C2CCC(CC)O2)=O)CC=CC(NC(c2csc(CO)n2)=O)C1 59906,c1(C(=O)NC2C(CNC(c3ccnnc3O)=O)CCC2)cccc2[nH]nc(O)c12 59907,C#Cc1cncc(C(N2CCCC2C2CCN(CCN3CCNC3=O)CC2)=O)c1 59908,C(=O)(CCC(C)(F)F)NCCCCC(C)NC(C(C)C)=O 59909,c1(Cc2cccc(CNC(C3(CC)CCC(O)CC3)=O)c2)ccccc1[N+](=O)[O-] 59910,C(=O)(C(C(C)C)NC(C)=O)N(CC(CN(C(CCN(S(CC)(=O)=O)C)=O)C)O)C 59911,c1(N(C)C)ccccc1C(N1CC(C)(NC(C2C3CC4C(C3)C24)=O)C1)=O 59912,c1(CC(C(=O)OCC)NC(=O)COCc2cn(CC)nn2)ccc(I)cc1 59913,C1(NC(C2C(C)(C)C2)=O)CC12CCN(C(c1ccn(CC(F)(F)F)n1)=O)CC2 59914,c1(C(N2CCC(C(C)NC3CC3)CC2)=O)ccccc1F.c1(N)nccc(C(=O)O)n1 59915,C12(CNC(Cc3nnn(-c4ccc(C)cc4)c3C)=O)CC=CCN1CCC2 59916,c1(NCCCOCC)ncc(S(=O)(=O)N2CCS(=O)(=O)CC2C)cc1Cl 59917,Cc1cccc(Cl)c1-n1cc(C(N2CCC(NC(=O)CCN(C)C)CC2)=O)nn1 59918,C(=O)(CC(C)CC(=O)OC)N1CCCC(CC(=O)N(CC(C)OC)C)C1 59919,c1(C(N2CC(n3ccnn3)C(O)C2)C(=O)NCC)ccc2c(c1)sc(=O)n2C 59920,CC(C)CC(C)(CNC(=O)Cc1ccccc1O)NC(c1n[nH]cc1I)=O 59921,C1(c2onc(-c3cc(F)c(O)c(F)c3)n2)CCC2(CCOCC2)CO1 59922,c1(NCCNC(=O)NC2C(C)CCN(S(C)(=O)=O)C2)cc(F)c(Cl)cc1O 59923,Cn1cnc2c(NC3CCN(Cc4ccc(Br)c(Cl)n4)C3)ncnc12 59924,C1(C(=O)OC)CCC(C(=O)NCC2CCCN(C(C3(C(C)(F)F)CC3)=O)C2)CC1 59925,C1(N(C(=O)CC2(NC(c3cc(F)n[nH]3)=O)CCCC2)CC)CCCN(C(C)=O)C1 59926,C1(CN(C)C(C2CCC(=O)N2C2CC2)=O)CCCN(C(=O)C=Cc2cc[nH]n2)C1 59927,c1(C(=O)NC(CCNC(C=CC(C)(C)SC)=O)C)ccn(C2CCC2)n1 59928,S(=O)(=O)(CC(=O)NCC1CN(C(c2cnc(Cl)n2C)=O)CC1O)NCC 59929,C1(C)(CNC(C(C)CN2CCOCC2)=O)CN(C(=O)C(=O)N(C)C)CCO1 59930,C1(COC)(CNC(=O)CC(C)F)CCCN1C(c1cccc[n+]1[O-])=O 59931,CCCC(CCC)C(=O)N1CCCN(C(=O)Cn2cccc(N)c2=O)C(C)C1 59932,C1(C(N(C(C(=O)OC)C)C)=O)C(C)OCCN1C(C1CS(=O)C1)=O 59933,S(=O)(=O)(C1CCCN(C2CC(=O)NC2)C1)Nc1c(CCOC)cccc1 59934,N1(C(c2cn(CCNC(c3c(COC)noc3)=O)nc2)=O)CCC(CO)C(O)C1 59935,N1(C(C(C)CO)=O)CC2(C1)CN(C(c1cn(C)cc1C(F)(F)F)=O)C2 59936,C1(C(=O)NCCOC)CC12CCN(C(c1ccsn1)=O)C2 59937,C1(c2n(CC=C)nnn2)(NC(C)(C)C2CC2)CC2CC1CC21OCCO1 59938,c1(CC(=O)NCC2(C)N(C(Cc3c(C)n(C)nc3)=O)CCC2)cc(F)ccc1Cl 59939,C(CNC(C1CC=CC1)=O)(C(C)C(C)C)NC(c1c(NCC)cccn1)=O 59940,N1(C(c2c(CC)n[nH]c2)=O)CCCC(N(CCO)C(c2ccoc2C2CC2)=O)C1 59941,Cc1nscc1C(=O)N(C(C)C(=O)NCc1nocc1C(C)C)C1CC1 59942,c1(C(N(C2CC(C(N3CCC(O)CC3)=O)C2)C)=O)ccc2occc2c1 59943,C12(CC(=O)NC3CN(C(=O)CCc4nc[nH]n4)CC3O)CCC(CC1)C2 59944,c1(NS(C2COC(C3CCN3)C2)=O)nc(Cl)cc(Cl)n1 59945,CCC1=C(C(=O)N2CCCCC2CCNC(=O)CC(O)CN(C)C)CCCO1 59946,N1(C(C(c2ccn(C)c2)C)=O)CCCC1c1ccsc1 59947,C(=O)(C(C(C)(C)C)NC(c1ccccn1)=O)N1CCN(C(CC)=O)CC1 59948,C1(C(=O)NC(CNC(c2c(C)ocn2)=O)(C)C2CC2)CCn2ccnc2C1 59949,c1(N(c2ncc(NC)cn2)C)ccc(N=c2ncnc3[nH][nH]c(Br)c2-3)c(F)c1 59950,C1(C(N(CCC=C)CC)=O)CC2(CC2)CN1C(c1cn(CCO)nn1)=O 59951,C1(NC(c2nc(C(C)C)sc2)=O)CC2(CCCCN2C(C2(O)CCC2)=O)C1 59952,C(=O)(C(F)(F)c1cncs1)NCC(C)NC(=O)C(c1ccc(Cl)s1)C 59953,N1(CC(N2C(c3ccc(C)cc3)CCC2)=O)C(=O)CN(C)C1=O 59954,Cc1nc(N2CCOCC2C(=O)Nc2cccc(S(=O)(=O)F)c2)nc2ccccc12 59955,C1(O)(C(=O)NC(C(C)NC(C(C)(C)NC(=O)OC)=O)CO)CN2CCC1CC2 59956,C#CCCN=C(NCCc1ccccc1C#N)NCc1ccn(C)c1 59957,CC1C(C)N(C(=O)CSc2nnnn2C)CCN1C(=O)C(=O)C(C)(C)C 59958,N1(C(COC(C)=O)=O)CC(NC(C2(C)CC=CC2)=O)CC12CCC2 59959,C(CC(C(=O)N1CCCCC1CCNC(=O)CCCn1ccnc1C)OC)OC 59960,c1(C(=O)NC2C(C)CN(C(C3CCC(C)CC3)=O)CC2)nc2ccccn2n1 59961,c1(C(=O)NC2CC(F)(CNC(c3cnco3)=O)C2)ccc(F)c(F)c1 59962,N1(C(CC2CC(OC)C2)=O)CC(C(=O)Nc2cc(C)cnc2O)CC(C)C1 59963,C(=O)(C1=CCCCO1)N1C(C(=O)NCC2CCCN(C)C2)CC1 59964,c1(C(=O)NCC(C)(C)CNC(C23CC4CC2C3C4O)=O)ccc2c(n1)CCCN2 59965,C(C1C(C(=O)NCC2(CN(C(=O)CC(C)O)C)CC2)C1(C)C)=C(C)C 59966,CC1(C)CNC(=O)C1NC(=O)C=CCNC(=O)Cc1ccc(F)cn1 59967,c1(C2(C(=O)NCC=CCNC(CCC(C)OC)=O)CC2)ccccc1C#N 59968,C1(C(=O)NC(CNC(C(C)=C(C)C)=O)(C)CO)C2COC(C)(C)OCC12 59969,c1(C(=O)NCCCC2(NC(=O)CSc3ccccc3)CC2)cc[n+]([O-])cc1 59970,C1(O)(CNC(c2c(C)cno2)=O)CCCN(C(C2(N3CCOCC3=O)CC2)=O)CC1 59971,C1(Nc2cc(NC(C(COC)(C)C)=O)ncn2)CN(C)C(C)(C)C1 59972,Cc1ccc(C)c(CCCC(=O)NCC#CCNC(=O)CNC(C2CC2C)=O)c1 59973,C#CC1(C(N2CCC(OC)C2C)=O)CCN(C(C2C(C)(C)C2(F)F)=O)CC1 59974,c1(SCC(=O)NC2CCC(CNC(C3(SCC)CC3)=O)C2)ccc(Cl)cc1 59975,C(C(=O)NC(CC)C(=O)N1CC(O)(CCO)C1)(C(C)C)SC 59976,C(=O)(C(C)(C)C)NCC(C)(C)CCNC(CN(C)CC=C(C)Cl)=O.OC 59977,c1(C(=O)NCC2(O)CCN(C(C(C)SC)=O)C2)coc2ccc(OC)cc12 59978,C(=O)(C1=C(Cl)CCOC1)N1CCC(CC)CC1C(N1CCC1(C)C)=O 59979,C12(C(=O)NCC(CCC)C)CCCC1CCN2C(c1cncc(C)c1)=O 59980,CC1(C)CCCN(C(c2cscn2)=O)C1CNC(=O)CSCc1ccccc1 59981,C1(NC(=O)COC2CC(NCCC(=O)N3CCCC3)C2)CCCC(F)C1 59982,C=C(C)CCC(=O)NC(CN(C(=O)C(C)(c1ccccc1)OC)C)(CO)CO 59983,CC1(C)Cc2cc(Br)ccc2C1NC(=O)Cn1cc(CN2CCC(C)(C)C2)nn1 59984,N1(C(CCN(C)CCO)=O)CCCN(C(=O)CC2COC(=O)C2)CC1 59985,C1(F)(C(=O)NC(C)CCCNC(=O)Cn2cc(C3CC3)cn2)CCCN(C)C1 59986,C(C(O)CC(=O)NCc1nonc1C)NC(c1cc(C(C)=O)on1)=O 59987,c1(CCN(CCc2ccc(C=C)cc2)C2CC2)ccc2c(c1)CCO2 59988,C1(OC)(CNC(=O)CSCC(C)C)CCN(C(=O)Cc2cnc(C)[nH]2)C1 59989,N1(C(c2ncn(C)c2)=O)CC2ON=C(CNC(c3ccc(NC=O)cc3)=O)C2C1 59990,c1(NC(C(c2csc(Cl)n2)N(CC(=O)OC)CC(=O)OC)=O)ccc(SC)cc1 59991,c1(OC)ccc(CN2CC3CC3(C(=O)Nc3cc(Cl)ncc3Cl)C2)cc1Br 59992,C1(C(=O)NC2(C(=O)NC(C)CC3CC3)CC2(C)C)C(C)(C)C1(C)C 59993,Cc1nc(C)c(CC(=O)NCC(C)(C)CNC(c2cc(C3CCCC3)no2)=O)s1 59994,C1(NC(CC=C)=O)CCN(C(c2ccnc(OC(C)C)c2)=O)C(C)C1 59995,N1(C(C(C)=C(C)C)=O)CC2CC(NC(=O)C(C(C)C)n3ccnc3)C1C2 59996,N1(C(c2scc(OC)c2)=O)CCCC(F)(C(N2CCC(C#N)C2)=O)C1 59997,Cc1c(F)ccc(C(N2CCN(C(=O)CCC(N)=O)CC(O)C2)=O)c1C#N 59998,c1(C(N(CCCCCC)CCNC(=O)C(C)(O)COC)=O)cc(F)c(F)c(Cl)c1F 59999,c1(C(N2CC(C(=O)Nc3ccnc(C)n3)C(O)CC2)=O)cc2cccc(O)c2[nH]1 60000,Cc1cc(F)ccc1Cn1nnnc1CC1(N2CCOCC2)CCCOC1 60001,CC1=C(C(=O)N2CCC(CNC(C3OCCC3(C)C)=O)C(C)C2)C(=O)OC1(C)C 60002,c1(CC)c[nH]c2cc(NC(C3C4CN(C(=O)C(F)(F)C(F)(F)F)CC34)=O)ccc12 60003,CC1(C(=O)NCCC(N)=O)CCN(Cc2ccncc2Cl)C1 60004,C1(CC(N2CC(O)(CN(C(c3cc(C(C)=O)oc3)=O)C)C2)=O)COCCOC1 60005,N1(C(CC)=O)CC2=C(C1)CN(C(=O)Cc1cnc(C3CC3)[nH]1)C2 60006,C(=O)(C(F)(F)C(F)F)NCC(CN(C(C1CCCC1C(F)F)=O)CC)(C)C 60007,C(CCC)(C(=O)N1CCC(CN(C(=O)CN2CCCCCC2)CC)CC1)=CCC 60008,N1(C(C(C2CC2)OC)=O)CCC(CNC(c2cnn(C(C)C)n2)=O)C(F)(F)CC1 60009,c1(N2CCC(C3N(C(CCCC(C)=O)=O)CCC3)C2)nc2cccnc2s1 60010,Cc1sc(Br)c(C(=O)NC2CC(F)CN(C(=O)C=CCO)C2)c1C 60011,CC1CN(C(C2(C#N)CC2)=O)CCN1C(=O)C(C)C(F)(F)F 60012,Cc1cccc2cc(C(=O)NC(C)CNC(=O)C(c3ccc(C#N)cc3)C)nn12 60013,C1(C)(C(=O)NC(CNC(c2nn(CC)c(O)c2)=O)CO)CC(C(F)(F)F)=NO1 60014,N1(C(CCCc2ncc(C)o2)=O)CCCC(NC(c2c(C)nc(C)n2O)=O)CC1 60015,Cc1ccc(C=CCC(=O)NC2(CCNC(C3CC3F)=O)CC2)cc1 60016,Cc1c(C(=O)NC2(C)CC(NC(=O)C(O)C(F)(F)F)C2)sc2nnc(S)n12 60017,N1(C(c2c(C)coc2C)=O)CCC(NC(c2cnn(C)c2C(F)(F)F)=O)C(F)C1 60018,c1(C(=O)NC(C2CCCN(C(c3cc(C(C)=O)on3)=O)C2)C)cccc(Cl)c1F 60019,c1(CC(=O)NC(CC)CN(C(C2CC2C)=O)CC)cc(=O)n(-c2ccccn2)[nH]1 60020,C1(NC(C2C(OC)C2)=O)CN(C(=O)CC2CC2)CC1c1ccnn1C 60021,N1(C(C2C(C=C)C2)=O)C(CNC(c2c[nH]nc2C(F)F)=O)CC2CCCC12 60022,CCC(C(=O)NC1(C2CCN(C(c3cccc(OC)n3)=O)C2)CC1)C(C)(F)F 60023,n1(CC(N2C(CN(C(c3n(C(CC)C)ncc3)=O)C)CCC2)=O)cccnc1=O 60024,c1(C(C(=O)NCC(CC=C)NC(=O)Cc2cccc(OC)c2)=O)ccc(O)cc1 60025,O=[N+]([O-])c1ccc(C(c2nnnn2C2COC2)NCCOCC2CC2)cn1 60026,C=C1CCCN(S(=O)(=O)CC)C1.C1C(C)C(=O)N1CC(C)C 60027,N1(C(c2c(NC)cccc2OC)=O)CC2(CC(N)C(O)C2)C1C(=O)OC 60028,CCC(C)(COC)C(=O)NCCC1(NC(=O)C(N)=O)CC1 60029,C1(F)(CNC(C2C(CC(C)C)C2)=O)CCCN(C(c2cc(N)ccc2O)=O)C1 60030,N1(C(C=CC(C)NC(C(C)OCCOCC)=O)=O)CC(F)(C(N)=O)C1 60031,Cc1cc(NC(=O)C(N2CCCC2CC(c2ccccc2)O)=O)c(C)s1 60032,N(C(=NCCc1ccc(F)cc1C)NC1CC1C)CC1(OCC)CCSCC1 60033,C(CCC(C)C(=O)N1CC(C)(OCC(=O)NC2CCC(=O)NC2C)C1)OC 60034,N1(C(c2cccc(OC)n2)=O)C2CCC1C(CNC(c1cc(C)cc(Cl)n1)=O)C2 60035,c1(SCCC(=O)N(CC(CN(C(C(C)(C)OC)=O)C)O)C)cc(F)ccc1F 60036,O=C(CCN=c1[nH]ccs1)NC1CC(NC(c2ccn(C3CCCCC3)n2)=O)C1 60037,N1(C(C23CCC(N=[N+]=[N-])C2C3)=O)C2CCCC1CN(C(=O)C=C1CCC1)C2 60038,C1(CNC(c2csc3nnsc23)=O)CC2CCC(C1)N2C(c1cscn1)=O 60039,c1(NC2CC(CC#N)C2)cc(Br)ccc1S(=O)(=O)N1CCSC(C)(C)C1 60040,c1(C(N2CCC(Cc3cn(CCC(C)C)nn3)C2)=O)ncc(Br)cc1Cl 60041,O=CN1CCCC1C(N1CCC(CNC(=O)Cc2cnco2)C1)=O 60042,c1(N(C)C(c2ccc(-n3cncn3)nc2)=O)nc2c(F)cccc2n1C 60043,Cc1ccc2ncnc(N(C(=O)CCC3CCC3)CC3CNCCO3)c2c1 60044,c1(C(N2CC(CC)(NC(=O)Cn3ccnc3C)C2)=O)cnc2[nH]cncc1-2 60045,C1(NC(C2(F)C(C)C2)=O)(CNC(=O)CCCOC(C)=O)CCCC1 60046,N1(C(C2C(C3(C)COC3)C2)=O)C2CCC(C(N3CCCC(F)(CO)C3)=O)C1CC2 60047,C(=O)(C(O)CC(F)(F)F)N1C(C(C)C)C(C(=O)NCC(C)Cc2cn[nH]c2)CC1 60048,c1(CN=c2c3ccc(OCC)cc3o[nH]2)cccc2c1CCN(C(C)=O)C2 60049,Cc1nc(C2CC2)ncc1C(=O)NCC1CCCCCN1C(=O)CNC=O 60050,c1(C(N(C2CCCNC2)CC)=O)ccc2c(c1)C=CC(C)(C)O2 60051,CN1CCN(C(=O)CC2CCCC(=O)N2)C(CNC(c2nccc(Cl)c2O)=O)C1 60052,C12(NC(c3ccc(OCC=C)cc3)=O)CCC(CC1NC(=O)CNC(N)=O)C2 60053,c1(CC)ccccc1C(C(=O)NC1CCCC1)N(n1ccnc1C)CCOC 60054,c1(OCC)cc(C(=O)NCC(CNC(C2(CC)CC2(F)F)=O)CO)ccn1 60055,c1(C(N2CCC(N(C(=O)COCC(F)F)CC)C2)=O)c(C)ccc(C)c1O 60056,C(CNC(C1CC1c1ccn(C)n1)=O)(CC(C)C)NC(c1nc(OCC)sn1)=O 60057,CC(C(=O)NCCC1(NC(c2ccc(C(C)(C)C)cn2)=O)CCC1)S(N)(=O)=O 60058,c1(C(=O)NC2CC(CNC(C3(COC)COC3)=O)C2)sc(C)c(C)c1C 60059,C(=O)(CCC(C)(C)NC(C12CSCC1C2)=O)NC(c1cn(C)cn1)C 60060,C1(CNC(CC(=O)NC)=O)COC2(COCCN(C(C3CC(=O)C3)=O)C2)C1 60061,C1(NC(=O)CCC2CCCO2)CC2CCC(C1)N2C(C1CCC2C(C1)C2(F)F)=O 60062,CC1CN(C(c2ncc(Cl)cc2F)=O)CC(C)C1NC(c1cnc(Cl)s1)=O 60063,N1(C(=O)COCC2(F)CC2)CC2CCC1(CO)C2 60064,N1(C(CN(C)CC)=O)CCC2CC1CN(C(=O)CCc1cnc3n1CCCC3)C2 60065,CC1(C)OC2CCN(C(=O)Nc3nccn4ccnc34)CC2O1 60066,Cc1cc(=NCc2nnc(CCO)s2)[nH]c(NC2CC2C(C)(C)C)n1 60067,Cc1nc(NC(c2ccc(-n3ccnc3C)cc2)C)cc(N(CC(Cl)(Cl)Cl)C)n1 60068,N1(C(c2ccc(CC)[nH]2)=O)CCOCCC1C(=O)NC(c1cc(C)on1)C 60069,c1(C(C(=O)NCC2N(CCc3nc(C)sc3)CCC2)(C)C)cc(F)cc(F)c1 60070,c1(CC)ccccc1CC(=O)NCC12CC1CN(C(C1CC(SC)C1)=O)C2 60071,C12(CNC(=O)C3=CCCCCC3)CCCC1N(C(c1cccc(O)n1)=O)CCC2 60072,c1(C(=O)NC2C(OC)CN(C(=O)C(C)(C)S(C)(=O)=O)C2)cnc2c(c1)CCOC2 60073,c1(C(N2CCC(C(O)C(F)(F)F)C2)C(=O)NCC)cncn1C 60074,C1(Cc2cn(CC(CNC(c3sccc3C(C)=O)=O)OC)nn2)C(C)(C)C1(F)F 60075,CN1CC2CC1CN2C(=O)CC1CN(Cc2cnc(Cl)nc2)CCO1 60076,C1(C(N2CC(CC=C)(C(=O)NCC(C)C(C)(F)F)C2)=O)CC2(CCC2)CO1 60077,C1(C(N2CC(C(C)OC)C2)=O)(COC)CN(C(=O)CC23CCCC2C3)C1 60078,C12(NC(c3nc(CC)sc3N)=O)CCC(CNC(=O)C(C)CN(C)C)(CC1)OC2 60079,C(=O)(C1(C)CCn2ccnc21)NC1C(C(N(CC(CN(C)C)O)C)=O)COC1 60080,C(=O)(CC(C)C(F)(F)F)N(C1(C(N2CC(CC)C(O)C2)=O)CC1)C 60081,C(CC)(CC(=O)N(C)CP(C)(C)=O)N(C(CN(CCC)C)=O)C 60082,C1(F)(CNC(=O)CCCc2nccs2)COCCN(C(=O)CC2COCCO2)C1 60083,N1(C(C(C)CC(F)F)=O)CC2(CCCC2NC(c2ccc(-c3cc[nH]n3)s2)=O)C1 60084,c1(C(C)C)scnc1C(=O)NCC(O)CNC(c1ncc(C(F)F)s1)=O 60085,C=C(C)CC(C(=O)NC1C2CCC1CC2)NC(C1CCN1CC)=O 60086,c1(C(=O)NC2CC(NC(CC(C)(C)OC)=O)C2)ccc(N(C)C)cc1F 60087,n1(CC(=O)NCC2C3CN(C(CC(=C)C)=O)CC32)cc(P(C)(C)=O)cn1 60088,Cc1ccc(C(N2CC(F)CC2C(N2CC3C(CN(C)C)C3C2)=O)=O)nc1C 60089,c1(CNC(CCOCCN(C(CC(C)CN(C)C)=O)C)=O)cccc2c1OCC2 60090,CC1CCCCC1(CNC(C1CC2CCC1O2)=O)NC(C1CCCC2(CC2)C1)=O 60091,c1(C2CN(C(=O)NC(c3nccn3CC(F)(F)F)CCC)C2)ccc(Br)cc1 60092,S(=O)(=O)(c1cnn(C2CCCC2)c1)N(CC=C)CCN(C)C 60093,N1(Cc2cccc(C)c2)Cc2ccc(C(=O)Nc3cncc(Cl)n3)cc2C1 60094,C1(C(=O)NC2(CC=C)CN(C(C3CC4CCC3CC4)=O)C2)CC2CCC1CC2 60095,c1(C(=O)NCC2CC(C)N(C(=O)C3CC3)C2)nc(O)nc(O)c1F 60096,c1(NC2CC(OC(C)(C)C)C2)nccc(=NCC2CCN(CC3CC3)C2)[nH]1 60097,N1(C(CC)C(=O)NC2CC3CC2N(C(=O)CSC2CC2)C3)CCc2ccccc21 60098,C(=O)(C(CCF)NC(=O)CCOC(C)C)N1C(C(=O)OC)CC1C 60099,N1(C(c2ccc(SC)cc2)=O)CC(NC(c2cc(Br)ncc2F)=O)C(F)(F)C1 60100,CC1(C)CCCC1(C)NC(c1cnc(CNC(C2CN3CCC2C3)=O)nc1)=O 60101,c1(C(C)(C)C)nc[nH]c1S(=O)(=O)NC12CC1CS(=O)(=O)C2 60102,c1(CNC2CCCC(C)C2)cc(Cl)c(Br)cc1F 60103,c1(N2CCC(CCC)C2)nc(N(C)CC2COC(=O)O2)nc2cc(C)ccc12 60104,C1(C(=O)NCCCCNC(C2(OC)CC2)=O)(N(C)C)CCCSC1 60105,c1(N2CCCC(CCCC)C2)nc(=NC)nc(N2CCOC(C(C)(C)C)C2)[nH]1 60106,N1(C(CCCn2cnc(C#N)n2)=O)CCC2CCN(C(=O)COC3CC3)C2C1 60107,C(=O)(C(F)C(F)(F)C(F)(F)F)N1CCCC(NC(c2ccc(COC)[nH]2)=O)CC1 60108,C(=O)(C(CCC(C)C)N=C1NS(=O)(=O)c2ccccc21)NCCNC(=O)NC 60109,c1(C(=O)NCC(CN(C)C(c2coc(Br)n2)=O)O)ccccc1S(C)=O 60110,c1(C(N2C(CNC(C(C3CCOCC3)OCC)=O)C=CC2)=O)cncc(Cl)c1C 60111,N1(C(CC(C)SC)=O)CC2(C1)OC1(C)CC2(NC(=O)C(C)Oc2ccccn2)C1 60112,C1(NC(C2(OCC)CCOCC2)=O)CCC(C)N(c2ncc(Br)c(C)n2)C1 60113,N12CCC(C1)CC(=O)N(CCCO)C(C)(C)C=CC2=O.C1(NSC)CCC1 60114,CC1(C)CCN(C(c2ncncc2Cl)=O)C1C(=O)NCCC1(O)CCCCC1 60115,C(=O)(C(CC)CC(F)F)N(C1(CC=C)CN(C(=O)CC(C)n2ccnc2)C1)CC 60116,C1(C(=O)NC(C2CCN(C(c3conc3C(C)(C)C)=O)CC2)C)CCS(=O)(=O)C1 60117,c1(OC)ccc2c(=NC(C)CCF)[nH]c(=NCc3ccc(Br)c(F)c3)[nH]c2c1 60118,Cc1cc(OCCC(=O)NCC2(F)CCCN(C(=O)CCC(F)F)C2)cc(C)c1 60119,C#CCC(C)(CNC(=O)CCCN(C)C(C1CC2CC2C1)=O)CO 60120,CC1SCCC1N=c1nc(N2CCCC(F)C2)c2c([nH]1)COC2 60121,Cc1ncc(C=CC(=O)NCC2COCCN2C(=O)COC2CC=CC2)s1 60122,c1(OC)c(C)ccnc1NC(=O)NCC1CN(c2nnnn2C)C1 60123,C(=O)(CC(=O)NC1C=CC(CNC(=O)C(F)CC2CCC2)C1)OC 60124,N1(CC)CC(C(=O)NCC2CCN(C(=O)C(c3ccc(Cl)cc3)(C)C)C2)CC1=O 60125,c1(C(=O)NCC(C(C)(C)C)NC(c2ccc3c(c2)CC3)=O)cc(O)nc(O)n1 60126,C1(N(C)CC2CC2)CCCN(N2CCC(OCCCC)C2)C1 60127,C1(C(=O)NC(C(=O)N(CCOCC)C)c2ccoc2)CCS(=O)CC1 60128,C=CCC(C(=O)NC1CCN(C(=O)C=C2SCC(=O)N2C)CC1F)C(C)(C)C 60129,C=CC1(O)CN(C(=O)C(C)N(C(=O)CC2CC3C=CC2C3)C2CC2)C1 60130,Cc1nc2ccc(C(=O)NC(C)CNC(c3cc4ncc(C)cn4n3)=O)cn2n1 60131,C1(CC(=O)NCC2C(C)CC2)CCN(C(=O)Cn2ccnc2)C1 60132,C1(C(=O)N2CC(SC)C2)CCCN1.C(=O)(CC(=O)OC)NC 60133,C1(F)(CNC(C=CCCC)=O)CCCN(C(=O)CCn2c(C)c(C)sc2=O)C1 60134,Cc1cncc(F)c1C(=O)NC1CCC(CCNC(=O)CC#N)C1 60135,C1(C(=O)OC)(CNC(=O)Cn2cc(CC3(C(F)(F)F)OCCO3)nn2)CCCO1 60136,C(=O)(CC(C)(C)C(F)(F)F)NCC1N(C(CCOC)=O)CCC1C1CC1 60137,c1(SC)ccc(C(=O)NC2CN(C(=O)CC3COC(C(F)(F)F)C3)C2)cc1 60138,CC(C)(C)CC(O)C(=O)N1CCN(CCNC(=O)C(c2ccncc2)O)CC1 60139,Cc1cc(C(=O)N(C)CCN(C(=O)C2=NOCC2)C)c2[nH]cnc2c1 60140,N1(C(C(C)=CC)=O)CC2(CNC(c3cn(-c4ccn(C)n4)cn3)=O)CCC1CC2 60141,CCC(CC)C(F)C(=O)NCC1(C)CN(C(C2CCCN2CC(C)C)=O)CCO1 60142,Cc1cc(C)c(C)c(C(N2CC(O)(C(C)NC(=O)CCc3cscn3)C2)=O)c1C 60143,C1(C(N2C3C(NC(C(CC)OC)=O)(CCC3)CC2)=O)CC2CC1C1C2C1(F)F 60144,C1(NC(Cc2cc(C)sc2)=O)CC(O)CN(C(c2c(O)cccc2F)=O)C1 60145,c1(CNCC(=O)NC23CC2C3)cccc(OCCF)c1 60146,C1(C)(NC(c2c(OC)oc(C)n2)=O)CCCN(C(=O)CCn2ccnn2)C1 60147,c1(OC)nc(OC)nc(N2CCC(C(N3CC4CCCC4C3)=O)C2)n1 60148,c1(C(N2CCC(NC(C(C)F)=O)C(F)C2)=O)ccc(Br)c2cccnc12 60149,C(CCC1CCC1)(C(=O)NOC1CC1)NC(CC(CC)OCC[Si](C)(C)C)=O 60150,C1(C(N2CCC(=C)CC2)=O)CN(C)CCN1C(=O)Cn1ccnn1 60151,c1(C(N)=O)cccc(C(N2CCOCC2CNC(=O)C=C2CCC2)=O)c1N 60152,C1(C(N2CC(CNC(CC=C=C)=O)C(O)C2)=O)COc2c(OCC)cccc2C1 60153,CCC(CC(=O)N(C)CCOCCOC)NC(=O)CC1CCOC1C 60154,c1(C(=O)NCC(n2cc(CCC(C)O)nn2)C)cc2c(O)cccc2s1 60155,C(CC(C)CCO)NC(c1cncc(C(C)(C)C)c1)c1n(CC(=C)C)nnn1 60156,N1(C(c2c(SC)scc2)=O)CCN(C(=O)CS(N)(=O)=O)CC12CC2 60157,c1(C(C)OCC)nc(C)c(C(N2CC3CC3(NC(=O)CCCOC(C)C)C2)=O)s1 60158,C=C(C)CCC(=O)NC(C1CCN(C(=O)C(C)N(CC(F)(F)F)C)CC1)C 60159,N1(C(C(C)OC)=O)CCC2CN(C(C3(O)CCC3)=O)CC2C1 60160,c1(C2(C(N3CC(CCNC(CCOCC)=O)C3)=O)CCCC2)cccc(Cl)c1 60161,C=C(C)C(CC(=O)N(CCC(N1CC2C(C1)C2(C)C)=O)CCO)OCC 60162,C1(C(=O)NC(c2nncn2C)C)CN(C(=O)CCc2cn(C)cn2)CC12CCC2 60163,C1(NC(CCc2c(OC)cc(C)cc2)=O)CCN(C2CC2)CC1C#N 60164,c1(CCC)cc(C(=O)NCC2COC(CNC(=O)CN3CCOCC3)C2)c(C)o1 60165,CC12CSCC1CN(c1ncncc1Br)C2 60166,c1(C(=O)NCC2CCCN(C(C=CC3(C)COC3)=O)C2)ccc2ccsc2c1 60167,c1(C(=O)OCC)nnc2n1CCN(C(C(C)=Cc1ccccc1)C(=O)NC)C2 60168,C1(C)(CNC(c2ccc(Cl)c(Cl)c2)c2n(CC=C)nnn2)CCS(=O)(=O)CC1 60169,c1(C(=O)NCCC#N)ncccc1NC(=O)Cc1ccc(C2CCC2)cc1 60170,c1(OCC)cccc(NC(=O)C(c2csc(Cl)n2)N(C)CCOC)c1 60171,C1(CC(=O)NC2C(CNC(=O)C=CCN3CC4CC4C3)COC2)CCCCCC1 60172,C(N=c1[nH]c2ncnc-2c(C(C)=O)[nH]1)C1OCCN(C(c2c(CC)ccs2)=O)C1 60173,C1(CC(=O)NCC2CCCC(F)C2)C2CN(C(C3CC34CCCC4)=O)CC12 60174,C(C)(C)(C#CCCC)NC(C1CC(CCNC(C(C=C)(C)O)=O)C1)=O 60175,C(C(C)(CO)NC(c1csc(CS(C)(=O)=O)n1)=O)NC(C(F)=C(C)C)=O 60176,C(=O)(C(C)(C)CN1CCCC1)N(C)CC1CCN(C(C2C(C)C2C)=O)C1 60177,C12(C(=O)NC(CC(=O)OC)C3CCCCC3)CC1CN(C(c1cncnc1)=O)C2 60178,N1(C(C(COC)C)=O)CCN(C(=O)Cc2ccc(Br)s2)C(CO)C1 60179,C(=O)(C(F)C(C)CNC(=O)CCC(C)(C)OC)N1CCC(OC)C1C(C)C 60180,C1(C)(C(=O)NC(C)CCNC(=O)Cc2cnoc2)CC1(F)Cl 60181,c1(OC)ncnc(C(=O)NCC2CC2NC(c2ccc(C(C)C)cc2)=O)c1F 60182,c1(C(=O)NC(CC)CNC(c2cc(Cl)n(C)n2)=O)c(O)nnc2c1CCC2 60183,c1(C(=O)NC2C(NC(c3ccc(C(N)=O)cc3)=O)C2)cccn2ccnc12 60184,Cc1cc(O)ccc1C(N1CCC(NC(c2cnsc2C)=O)CC1C1CC1)=O 60185,C1(NC(C(C)OC)=O)CN(C(=O)CCS(=O)(=O)N(C)C)C(C)(C)C1 60186,C(=O)(CCC(=O)NCC1OCCC1C(=O)NC1(c2ccccn2)CC1)N(C)C 60187,C(CC(C)(C)C)(C(=O)NCc1c[nH]nc1C(=O)NOC(C)C)OC 60188,C1(NC(C=C(CCC)CCC)=O)CCC2CN(c3ncc(C)c(SC)n3)CC2C1 60189,C(C(CC(C)C)C(=O)NC1CC(CNC(C23CCC(N=[N+]=[N-])C2C3)=O)C1)OC 60190,CC(C)C(S(=O)(=O)N1CCC2(CC2)C1)c1ccccc1 60191,N1(C(c2c(C)ccc(C)c2)=O)CC2CC1CN(C(c1cnn3cccnc13)=O)C2 60192,c1(C(=O)NCCCCC2CN(C(Cc3cc(C)ns3)=O)C2)cc2n(n1)CCCC2O 60193,CCCCC(C(=O)NCCNS(C)(=O)=O)NC(c1cnn(C)c1)=O 60194,CCC(C)(COC)C(=O)N1CCN(CCNC(=O)C=CS(C)=O)CC1 60195,N1(C(CCC#C)=O)CC=C(C(C)(C)C(=O)NC(C)C(=O)NCCF)C1 60196,C(CNC(=O)C(C)(C)NC(C)=O)(CC(=O)N=c1ccn(CCCO)[nH]1)OC 60197,C1(CCNC(c2c(COC)ccs2)=O)COCCN1C(=O)CC1CCC(C)(C)C1 60198,c1(C(N(CC(C)NC(c2c(O)ccc(C)n2)=O)C)=O)cnc2c(c1)OCC(=O)N2 60199,C(CNC(C1CC2CC2C1)=O)(C(=O)N=c1cc2n([nH]1)CCCC2)N(C)C 60200,C(C(=O)N(CC(O)CN(C)C(c1nncs1)=O)C)(C1CCOC1)OCC 60201,CC(C)CC(C(=O)NCC1CCOC1(C)C)NC(=O)CCC(F)(F)F 60202,CC1(C)OC(=O)CC1C(N1CC(F)(CNC(=O)CC2NC(=O)NC2=O)C1)=O 60203,C1(C(C)C)CN(C(c2ccns2)=O)CCN1C(c1c[nH]c(=S)cn1)=O 60204,N1(C(c2cnn(CC)n2)=O)CCC(C2CC2NC(=O)C(C(C)C)NS(N)(=O)=O)CC1 60205,C(C(C)(C)C(=O)NC1CCC(CNC(=O)CC2CC2(C)C)C1)N(C)C 60206,C1(C2CC2)(C(=O)NC2CCC(NC(c3c(C)nc(CCCC)s3)=O)C2)CC=CC1 60207,c1(CC(N2CCC(NC(C(COC)C)=O)C23CC3)=O)cnc2n1CCOC2 60208,CC1C2CCN1NC2=O.N1(C(C2CC23CCC3)=O)CCC(O)CC1 60209,C(=O)(CCCC(C)(C)C#N)N1C(C(=O)NCc2c(CC)onc2C)C(CC)CC1 60210,c1(C2(C(=O)NC3C(NC(CSCCC)=O)C3)CC2)ccccc1Cl.C1CN1 60211,O=C(C1CCSc2ccccc21)NC1CCCN(C(=O)Cc2cnccn2)CC1 60212,c1(C(=O)NCCCN(C(c2cncc3nc[nH]c23)=O)CC)n[nH]c2c1NCCC2 60213,N1(C(CCC(C)C#N)=O)CC2(C1)OC1(C)CC2(NC(c2c(Cl)cnn2C)=O)C1 60214,CC1(C(=O)NCCCN(C(=O)Cn2ccnn2)CCO)CCCS1(=O)=O 60215,Cc1cnc2nc(C(=O)N(CC(C)(C)CNC(=O)C=CC3CCCO3)C)nn2c1 60216,N1(C(=O)NC2CC2)CC2CC2(C(N(c2cn(C3CC3)cn2)CCN(C)C)=O)C1 60217,C1(C)(CC)C=C(C(=O)NCC(C)CC(=O)N2CC(N(C)C)C(C)C2)C1 60218,CC1NC(=O)OC12CN(C(=O)CCOCCCNC(=O)CCc1ccccn1)C2 60219,N1(C(CCCCOCC)=O)CCC2(CC(NC(=O)C(C)OCC(C)C)C2)C1 60220,c1(C(=O)Nc2c(C)c(Cl)ncc2)cc2cc(-c3ccc(N(C)C)nc3)cnc2[nH]1 60221,c12cc(ccn1)CNC2=O.n1(C(C)C)cc(CC(=O)O)nn1 60222,C1(C(=O)NCC(N(C(=O)CCn2cccn2)C)C2CC2)CC12CCOCC2 60223,c1(NC(C2(C)CCN2C(C2(C)CCOCC2)=O)=O)cc(Br)ccc1CO 60224,CCC(CC)(CO)C(=O)NCCC1CN(C(C2CCCCC2F)=O)C1 60225,CCCC(CC)C(=O)N(C1CCCN(C(c2cc(O)nn2C)=O)C1)CCO 60226,N1(C(CCc2c[nH]c(=N)[nH]2)=O)CCCC(NC(C2CCNC2=O)=O)CCC1 60227,O=C1CCC2(CCCN(C(=O)Nc3cccc(CCO)c3)C2)CN1 60228,O=C(CCCCCCNC(C1CCCC1)=O)NCC1CCC2(CC2)CO1 60229,N1(C(C(C(C)C)C2CCC2)=O)CC(C(N2CC(N(C)C)C(C)C2)=O)C(F)(F)C1 60230,CC1CN(C(c2c(C(F)F)cnn2C)=O)CCCN1C(C1CNC(=O)N1C)=O 60231,C1(NC(C2N(CC)CC2)=O)CCC(N(C)C(C2(C)CC(C)=NO2)=O)CC1 60232,N1(C(Cn2c(=N)nc[nH]2)=O)CCCC(C2(NC(=O)COCC3CCOC3)CC2)C1 60233,C(C(C)C(=O)NC1CC(CO)C1)N(C(C(C)C)=O)C 60234,C1(NC(CC(C)(C)NC(CN(C)C)=O)=O)CCN2CCCCC12 60235,c1nc2ccccc2cc1C(=O)NCC1(CO)CC1.N1(OC)CCC2(C1)CN(C)C2 60236,c1(CC)cc(C(=O)NC2CC(CNC(C3CCOC(C(C)C)C3)=O)C2)ncn1 60237,CC1CN(C(C2(CNC(c3cc(Cl)no3)=O)CC2)=O)CCC1Nc1ccccc1 60238,C1(C)(C(=O)NCC(C)(C)NC(C2CCCCC2O)=O)CCC(=O)N1 60239,c1(C(=O)NC2CCC(N(C(=O)CCC3CCCCC3)C)C2)ccn2nccc2n1 60240,c1(CC)c(C(=O)NC(CNC(=O)C2CC2)(CC)CC)cnn1CC(C)C 60241,C1(F)(C(=O)NC2CC(N(C(CCN(CCC)C)=O)C)C2)CCOC1 60242,N1(C(CC2(OC)CN(C(c3cn(C)c(C)n3)=O)C2)=O)CC2(CCC(=O)N2)C1 60243,c1(CN2C(C(=O)NC(CNC(CCCC)=O)C)CCC2)cccc(Cl)c1 60244,C1(C(=O)NC(C2(O)CN(C(C34CC(F)(C3)C4)=O)C2)C)OCCOC12CCC2 60245,C1(CN(C)C(C23CC(F)C2C3)=O)CCCN(C(c2cnccc2Br)=O)C1 60246,c1(C(N2CC(C)NC(=O)C2)=O)ccc(S(C)(=O)=O)cc1F 60247,C(=O)(C1=CS(=O)CCC1)N1CC(NC(c2cc(CC)nc(O)c2)=O)C(CO)CC1 60248,C1(CNC(c2cc(CF)on2)=O)CN(C(C2(O)CCSCC2)=O)CC12CCC2 60249,C1(CNC(=O)CCCF)CCCCN(C(c2cc(Cl)cc(C(F)(F)F)n2)=O)C1 60250,C1(CNC(CN(C2CC2)CC)=O)CN(C(=O)CCC#N)CC(C(F)(F)F)O1 60251,c1(C(=O)NC2CC(C(C(=O)NCCCCSC)F)C2)nocc1Cl 60252,c1(C(=O)NC(C)CCN(C)C)n[nH]cc1-c1ccccc1 60253,c1(C(=O)NC(c2cccnn2)C)csc(CCN)n1 60254,c1(C(=O)NCC2(F)CC(CNC(C(C)N(C)C)=O)C2)ccc(SC(F)(F)F)nc1 60255,C1(CNC(=O)CCC2OCCO2)CN(C(=O)CC2=NNC(=O)C2)C2(CCC2)C1 60256,N1(C(Cc2ccc(C)s2)=O)CC=C(C(=O)NCC2COC(=O)N2)CC1 60257,C(=O)(C(C)CCCCCC)NCc1occ(C(N2C(C)(CCC)CC2)=O)c1 60258,C1(CNC(c2c(SC)cccc2)=O)CCCN(C(=O)Cn2nc(C)cc2C)CC1 60259,c1(C(N(CC(C)O)CCNC(C2C(OC)CC2)=O)=O)cocc1C 60260,C1(CC(=O)NC2(C)CSC2)CCCCC1NC(=O)CC1C(C)(C)C1(C)C 60261,N#Cc1ccc(CN2CCC(C(=O)Nc3ncccc3I)C(O)C2)c(Cl)c1 60262,N1(CC(N2CC(N(C(CC(C=C)C)=O)C)C2)=O)CCCCC(O)C1=O 60263,C(=O)(CC(C)(C)CC(F)(F)F)NC1(CO)CN(C(Cc2ccc(C)s2)=O)C1 60264,c1(OC)ccc(C(=O)NC2CC(NC(c3cnc(O)s3)=O)C(O)C2)c(N)c1 60265,C#CCC(C)(C(=O)NC(CO)CCC=C)NC(=O)C(C)C#N 60266,c1(CCNCc2c(CNc3c(C)cccc3)cnn2C)c[nH]c2cc(F)ccc12 60267,c1(C(N2C(CNC(c3cc(CC)[nH]n3)=O)COCC2)=O)cnn2ccnc(N)c12 60268,S(=O)(=O)(c1ccccc1Cl)N1CC(CN(C(C(N2C(C)CCC2C)C)=O)CCO)C1 60269,CC(C)C(C(=O)N1CCCC(CC(=O)NCc2ncccn2)C1)N(C)C 60270,n1(CCN(C(=O)CC2CC(C)(C)CO2)C)ncc2ccccc12 60271,c12ccc(c(I)c1)[nH]c2=O.C1(C)(C(=O)OC)C=CCN1C(C)=O 60272,C(=O)(CC1=CCOCC1)NC1C(CNC(CCOc2cc(C)cc(C)c2)=O)CC1 60273,c1(OC)ccc2c(=NC3CCCN(C)C3C)[nH]c(=NCCCCC#N)[nH]c2c1 60274,C1(C(N2CCC(N(C(=O)CC3CC=CC3)C)C2)=O)CCC(=O)N(C2CC2)C1 60275,Cc1cccc(C(N2CC(CC(=O)NC3(CC4CCC4)CC3)CC2C)=O)c1 60276,CC(C)(CC#N)C(=O)NC1COCCN(C(c2c[nH]nc2Br)=O)C1 60277,c1(C(=O)NCC2(C(N)=O)CN(C(C(=O)N(C)C)=O)C2)ccc(C2CCC2)nc1 60278,C1(C(=O)NCC(C)N(C)C(C2(CC3CC3)CCC2)=O)CC2(CC(=O)C2)C1 60279,CCCCCCC(F)C(=O)N(C)CC1(O)CN(C(=O)CC(C)(C)c2cccs2)C1 60280,CC(CO)C(C)N=c1nc(N(CC(F)(F)C(F)(F)F)C)c2c([nH]1)COC2 60281,CC1(F)CC2(CN(C(C3CCCN3C(=O)C(CO)C(C)(C)C)=O)C2)C1 60282,C1(CNC(C(C)NC(N)=O)=O)(NC(=O)CC2CCCCC2)CCCCC1 60283,C1(CNC(C(=O)NCCNS(C)(=O)=O)=O)CC2(CCNC2)CO1 60284,C1(F)(C(N(C)CCNC(C2CC23CCC3)=O)=O)CCCN(C(=O)OC(C)(C)C)C1 60285,Cc1cc(N(C2CCN(C(=O)C(O)CCc3ccccc3)C2)C)nc(C)c1C#N 60286,C12(NC(CN3CC(C)(C)C3)=O)CCC(CC1NC(c1cnn[nH]1)=O)C2 60287,C1(CNC(c2snnc2C2CCC2)=O)CCCN(C(=O)CC2CC2C2CC2)CC1 60288,c1(CN2CC3N(C(c4cc(Br)ccc4F)=O)C(C3)C2)c(F)ccc([N+](=O)[O-])c1F 60289,C(CCCOC)(C(=O)NCC(C)(C)COC)NC(C=CC(=O)OCC)=O 60290,CCCC(C)(C)CNC(=O)CC1CC1CNC(=O)CCc1ccc[nH]1 60291,C(CCC(C)(C)NC(C1CCCCCC1)=O)NC(C1(CC)COC1)=O 60292,c1(C(N(C2CCCN(C(c3n[nH]cc3[N+](=O)[O-])=O)C2)C)=O)ccc(S(C)=O)cc1 60293,c1(CNc2cn(CC(=O)OCC)nc2)c(OC)cc(Cl)cc1O 60294,c1(C(=O)NCC(N2C(C)C(C)(C)CC2)=O)n[nH]c2cc(Br)ccc12 60295,n1(C(C)C)cc(C(=O)NCC(C(C)(C)C)NC(c2cn(CO)nn2)=O)ccc1=O 60296,CC1(C)CC(C(=O)NC(CNC(C2CCS(=O)CC2)=O)CO)CNC1=O 60297,S(=O)(=O)(c1cn(C2CC2)nc1C)NC1CCN(C(CN(CCC)C)=O)CC1 60298,N#Cc1ccc2c(c1)CC(NC(C1CNCC(F)(F)C1)=O)C2 60299,C#CCC(CC(F)F)C(=O)N1CCC(N(C(c2cnc3cccnn23)=O)CC)C1 60300,c1(C(N2CC3C(CNC(c4c(C)n[nH]c4)=O)(C3)C2)=O)cnc2snc(C)c2c1 60301,N1(C(CSCC#C)=O)CC(CNC(C2CCCN2C(=O)NC)=O)CC1(C)C 60302,N1(C(C2C(C(C)C)OCC2)=O)CCCC2(C1)CN(C(c1ccnc(Cl)c1N)=O)C2 60303,C1(C(=O)NCC2CC(O)C(O)C2)CCCCCN1C(C1CC1Cl)=O 60304,c1(OC)cc(-c2noc(COC(C3CCC3)=O)n2)cc(Cl)c1OC 60305,N1(C(C2CC(OCC)C2)=O)CC2CCC(C1)N2C(C1Cc2nncn2C1)=O 60306,c1(CCC(=O)N(C(C)C(=O)N(CCCCOCC)C)CCC)nccn1C 60307,O=C1CC2OCCC2(C(=O)NC2CCCC2NC(c2cnc(S)nc2)=O)CN1 60308,c1(CCC(=O)NC(C(CO)NC(CC(=C=C)C)=O)C)ccc(Br)c(C)c1 60309,CC1CCN(C(=O)Cn2ccc(=N)[nH]2)C1CNC(=O)CCN1CCCCCC1 60310,c1(OC)noc(C)c1NC(=O)C(c1ccccc1)NC(=O)CC1CCCC12CC2 60311,N1(C(CC(=O)NCC)=O)CCC2(CC1)CC2NC(C1C=CCS1)=O 60312,C(=O)(C1CCCn2cncc21)N1CC(CNC(C(CCCC)O)=O)(COC)C1 60313,C1(C)(C(=O)OC(C(=O)NC)C)CC(C(C)C)=NO1 60314,C(C)(CCCCNC(C1CCOC1(C)C)=O)NC(c1ccc(CCCCCC)s1)=O 60315,N1(C(C)C(=O)NC(C)C(=O)Nc2ccc(Cl)cc2)Cc2ccccc2C1=O 60316,CN1CCC(C(=O)NCC2(F)CCN(C(c3ncncc3Cl)=O)CC2)S1(=O)=O 60317,CC1(C)COC(CC(N2CCCCC2CCNC(=O)CNS(C)(=O)=O)=O)C1 60318,N1(C(C2OCCN(C(C(CC=C)C(C)C)=O)CC2)=O)CCC2(CNC(=O)C2)C1 60319,C1(NC(C2N(C(c3cccc(C)n3)=O)C3(CC2)CC3)=O)CCc2ncnn2C1 60320,C1(NC(c2cc(OC)n[nH]2)=O)C2CC1CN(C(=O)C(F)CC1CCCCC1)C2 60321,C12(CNC(C=CCCC)=O)CC(NC(=O)C(C)C(F)(F)F)(C1)C1(CCOCC1)O2 60322,c1(COC)cc(CC(=O)N(C)CCN(C(=O)CC2CCC2OC)C(C)C)n(C)n1 60323,C(=O)(C(CNC(c1ccc2ccoc2c1)=O)CC(C)C)N(C(CCCC)C)C 60324,CCC(CNC(=O)CCP(C)(C)=O)(CC)C(=O)NC1CCC1(C)C 60325,C1(NC(c2n(CC)ncc2Cl)=O)CN(C(c2c(Br)n[nH]c2C)=O)CC12CC2 60326,N1(C(CCc2cc(OC)no2)=O)C(C)C2CC1C2NC(=O)C(CO)N(C)C 60327,N1(C2CCCN(C(C=CSC)=O)C2)CCN(C(=O)C(C)OCC(C)C)CC1=O 60328,N1(C(CC2OCCN(C(COC(CC)CC)=O)C2)=O)CCOC(C2CC2)(CC)C1 60329,C(=O)(C(CC)CCCCCC)N1CCC(NC(CC(=C)C)=O)(COC)CC1 60330,c1(C(=O)NCCC2C(C)CN(C(C3CCCC3)=O)C2)c(F)ccc2cnn(C)c12 60331,N1(C(=O)OCc2cc(OC)c(C)cc2)CC2CC(C)N(C(=O)C3CC3)C2C1 60332,C#Cc1ccc(CC(=O)NCC2(CC)CCCCC2)cc1.C12CC1CC(=O)N2 60333,C1(NC(c2cncc(Br)c2)=O)CC2(C1)CC(C(=O)NCc1cnco1)C2 60334,c1(OC(COC(C)=O)C(=O)NC(C2CCC(=O)NC2)=O)cc(C)cc(C)c1C 60335,N1(C(C2(CNC(C(CCC)C(C)C)=O)CCCO2)=O)CCc2nnnn2CC1 60336,C1(C(N2C(CNC(C(CC(C)C)O)=O)C=CC2)=O)CCc2ccccc2CC1 60337,c1(NC(C2CNCCN2Cc2ncccc2[N+](=O)[O-])=O)cc(Cl)c(O)c(Cl)c1 60338,N1(C(C(CC)(C)C)=O)CCC2(CC1)CC(NC(c1cc(SC(F)(F)F)c[nH]1)=O)C2 60339,C(C(O)C(=O)NC1(C(=O)N(C)CCO)CCC1)OC 60340,c1(NCCOCCNC(C(C)(C)N(C)C)=O)cc(C#N)ccc1[N+](=O)[O-].C1CO1 60341,c1(NC(C2CC(F)CN(Cc3cc(Br)ccc3I)C2)=O)cnc2ccc(F)cn12 60342,CCC(C(=O)N1CCC(CNC(c2csc(CC(F)F)n2)=O)C12CC2)C(F)(F)F 60343,c1(C(C)(C)C)ccc(C(=O)NCCOC2CN(C(=O)CCC3CC3(C)C)C2)[nH]1 60344,c1(C(=O)Nc2ccc(C)c(F)c2)cc2c(nc1N)CCC2 60345,C1(CC(=O)NC(C)CCNC(=O)CCn2ccnn2)C2CC3CC(C2)CC1C3 60346,C1(CNC(COc2cc(C)on2)=O)CN(C)CCN1C(C1CCCN1C1CC1)=O 60347,N1(C(C2(CC#C)CCCC2)=O)CC2CC1CN2C(=O)C(C1CCS(=O)(=O)CC1)O 60348,C(C)(C(=O)NCCN(C(=O)CCC1CCCO1)C)NC(=O)NC 60349,C1(OC)C2CC3CC1CC(C(N1CCC(NC(=O)C(=O)N(C)C)C(F)C1)=O)(C3)C2 60350,c1(C(=O)NCCC(=C)CNC(=O)C(C)CC=CC)c(C(F)(F)F)cccc1Cl 60351,C#CC1(C(=O)NCC2CC(C(=O)N3CCS(=O)(=O)CC3)=NO2)CCCCC1 60352,C1(N(C(=O)C(O)CC2CCCO2)C)CCN(C(=O)C(C)(C)c2ccccn2)CC1 60353,c1(CCC)cnnc(C(=O)N(CCN(C(c2cc(OC)ns2)=O)CC)CC)c1 60354,c1(C(=O)NC(CCC)CNC(=O)C(N2CCCC2)C2CC2)cn(CC)nc1C 60355,C1(OC)NC(C(=O)NCCn2cc(CN3CCNC3=O)nn2)CCC1Br 60356,N1(Cc2c(OC)ccs2)Cc2[nH][nH]c(=NC(=O)c3ccc(F)c(O)c3)c2C1 60357,N1(C(C(C=C)(C)O)=O)CCC2(CC1)OCCC2NC(=O)C(C)CCOC 60358,N1(C(C=CCC)=O)CC2CC1CN(C(=O)Cc1cc(C)[nH]n1)C2 60359,N1(C(C(C)COc2ccccc2)=O)CCC2CCC(C1)N2C(=O)CCC(F)F 60360,N1(C(=O)OC(C)(C)C)CCC(C)(O)C(C(=O)NC2C3CC4C(=O)OC2C4C3)C1 60361,CCC(C)CCC(=O)NC(CNC(=O)CC12CNC(=O)C(C1)C2)CC 60362,N1(C(C(CCCC)NC(N)=O)=O)CCN(C(=O)C=Cc2ccsc2)CCC1C 60363,Cc1cc(Cl)cc(C(=O)N(C)CCNC(c2ncc(Cl)cc2Cl)=O)c1N 60364,C(=O)(C(C)C(F)(F)F)NCC(C(=O)NC(C1CCCC1)CC)C 60365,Cc1nccnc1C(=O)NC1COCC1NC(C1CC(C)(C)CO1)=O 60366,C(C)(C(O)C(=O)N(CCCNC(=O)C(N)=O)CC1CCCC1)SC 60367,c1(C(c2n(CC)nnn2)Nc2cccc(SC)c2)cc(Cl)c(Br)cc1F 60368,c1(OC)ncc(Br)cc1CN1CCCN(C(c2ccn(C(F)F)n2)=O)CC1 60369,N1(C(c2ncc(C)nc2)=O)CCC2(CC1)CC2(CO)CNC(=O)Cc1cocn1 60370,C1(C(=O)NCC(CNC(c2c(CC)scc2)=O)(C)C)CCC(N(C)C)CC1 60371,C1(NC(C(OC)OC)=O)CS(=O)(=O)N(C)C12CCN(C(=O)CC1(C)CCC1)CC2 60372,c1(OCCC)cccc(C(=O)NCc2cnsn2)c1 60373,C1(C(=O)NCC(C)(O)C2(C)CC2)CCCN1C(C1(c2ccccc2)CC1Br)=O 60374,c1(C(=O)NC(C(C)NC(c2csc(CO)n2)=O)C)ccccc1Br 60375,C(CCCN(C(=O)C=CC(=O)NC1CC1)C)NC(C1C(C(=O)OC)C1)=O 60376,C(=O)(CC(C)(O)C(F)(F)F)N(C1CC2N(C(C(C=C)(C)O)=O)C(CC2)C1)C 60377,N1(C(COc2cn(C(C)C)nc2)=O)CC(C)(C)OC2(CCOC2)C1 60378,C1(CCNC(c2c(C)occ2)=O)CN(C(c2cocc2Br)=O)CCO1 60379,c1(C(N(c2cccnn2)CCC)C2CC2)cc(CO)ccc1Cl 60380,Cc1ncc(C(N2CCC(NC(C3C4CNC(=O)C34)=O)C2)=O)cc1C#N 60381,C1(CN2CC(NC)C(O)C2)CC2(CCCO2)C1 60382,N1(c2nccc(OCCC)n2)CC2(CCC(NC(c3ccc(O)cc3)=O)CC2)C1 60383,N1(C(CS(=O)(=O)NC)=O)CC2CCCC(NC(=O)C(O)C3CCCC3)C2C1 60384,N1(C(c2c(C)ccs2)=O)CC2CCN(C(=O)C(c3ccc(Cl)cc3)O)CCC2C1 60385,CS(=O)(=O)c1cccc(-c2nc(-c3n[nH]cc3Cl)n(CC3CC3)n2)c1 60386,C1(CNC(c2n(C)cnc2)=O)C2CC2CN1C(c1cncc(O)c1)=O 60387,c1(OC)ccc(O)c(NC(=O)CCC2CCN(C(=O)CCCC(=O)N(C)C)C2)c1 60388,C1(CC)C(C(=O)NCCc2cccnc2C)CCN1C(=O)C(=O)NC1CC1 60389,c1(OC)cc(F)c(Br)cc1C(=O)NCC(O)CNC(=O)C=Cc1cnc[nH]1 60390,Cc1c(C(N2CC(O)(CC(N3CC(OCC(C)C)C3)=O)C2)=O)ccn1C 60391,N1(C(Cc2c(C)non2)=O)CC(C(N2CCN(C)CC2)=O)C(C2CC2)C1 60392,CC1CCN(CCC(=O)NC(C)(C)C2(C3CCCN3C(CC(C)(C)C)=O)CC2)CC1 60393,C=CCN=C(NCC(=C)Cl)NCc1csc(COCC)n1 60394,CC1CCN(C(c2c(C#N)ncn2C)=O)CC1CC(=O)N(C)CCO 60395,C(=O)(C1=C(C2CC2)N(C2CC2)C(=S)NC1c1cn2ccsc2n1)OC 60396,c1(C(N(CCNC(C(C(CC)O)C)=O)CC)=O)cc2ccc(Cl)cc2[nH]1 60397,c1(C(N2CC(CNC(c3nc(C)oc3)=O)C(C)C2)=O)cccc2occc12 60398,N1(C(c2c(CC)cno2)=O)CC2CCC(NC(=O)CCc3ccc(C)s3)CC2C1 60399,C=CC1(CC(N2CC(C)C2)=O)CN(C(S(C)(=O)=O)=O)C1.C1(C)(N)CCOC1 60400,C(N=c1nc2sccc2c(N2CC3CCC3(C)C2)[nH]1)CCc1ccn(C)c(=O)c1 60401,Nc1c(C(N2CCCC(CNC(c3cc(Cl)nnc3Cl)=O)C2)=O)nc(O)nc1O 60402,C1(NC(C=CCN(C)CC)=O)CCC(C(=O)NC2(CO)CC(F)C2)CC1 60403,Cc1c(C=CC(N2CCC(C)C(NC(c3c(Cl)cncc3Cl)=O)C2)=O)cnn1C 60404,c1(C(=O)NCCC(C(C)C)NC(C(C=CC)O)=O)ccc(Cl)c(F)c1 60405,c1(CC)[nH]nc(C(=O)NC2CCCCCC2NC(=O)CC(C)C)c1[N+](=O)[O-] 60406,C(CCN(C)OC)NC(C1(C)CN(C(C(CC2CC2)OC)=O)C1)=O 60407,CN1CCN(C(c2cnc[nH]c2=N)=O)CC1C(=O)NC1(C)CCCC1O 60408,c1(C(=O)NC(C)C(=O)N(C)C)ccc(SCCOC2CCOC2)cc1 60409,c1(CNC(CCCC#CC)=O)ccc2c(c1)CN(C(c1cccc(Cl)c1C)=O)C2 60410,C1(C)(C(N(CC)Cc2ccoc2)=O)CC(O)CN1C(=O)CC1CCCC2CC12 60411,CCC(Cc1ccccc1)CC(=O)NC(CNC(=O)CC1(O)CCOCC1)CC 60412,C1(C(=O)NCC(c2ccccc2)NC(C(C)Nc2csc(F)c2)=O)SCCCS1 60413,c1(CN2C(C(=O)NC(c3cnccn3)C)CC(O)C2)cc(Br)ccc1Cl 60414,c1(C(=O)NCCOC(C)=O)cc(Cl)ccc1C.C12(CC1)C(=O)N(C)CCOCC2 60415,c1(CNCCN(C(C2(CC)CCOC2)=O)Cc2ccc(F)cc2)coc(C#N)c1 60416,N1(C(C2OCC3CCCC23)=O)CCC2(CCN(C(c3cc(O)ncn3)=O)C2)C1 60417,C(=O)(C1CCCc2ncccc21)NCC(CNC(c1cn(CC(N)=O)nn1)=O)F 60418,c1(C(=O)NCCN(CCO)CC)ccc(C(=O)NC)cc1 60419,Cc1c(C(N2CC=CC2C(=O)NOC(C)C)=O)cccc1C#N 60420,C1(NC(CC2CN(C)C2)=O)CC2(CCN(c3ccc([N+](=O)[O-])c(O)n3)CC2)C1 60421,C=CCCCC(C)NC(C1(N(C(=O)C=CC(=O)N(C)C)C)CC1)=O 60422,C(C(C)(C)CNC(C1(O)CCCC1)=O)N(C(=O)CC(C)NC(C1CCCC1)=O)CC 60423,N1(C(c2cc(C)sn2)=O)CC(C(=O)NCC2(C)CC=CCC2)C2(CC2)C1 60424,C12(NC(=O)Cc3ccc(Cl)s3)CCCC1CN(C(c1cccc3c[nH]nc13)=O)C2 60425,c1(COC(N(CCCC(=O)NCC(CCC)C)C)=O)ccc(F)cc1 60426,N1(C(c2cc(C(C)(F)F)on2)=O)CC(NC(c2ccnc(O)c2)=O)CC(F)C1 60427,c1(C(N(C(CNC(CC2C(C)=NNC2=O)=O)C)C)=O)ccc2c(c1)CCC2(C)C 60428,N1(C(C=NOC)=O)CCC2(CC1)OCCC2NC(C1CC1c1ccccc1)=O 60429,c1(C(N2C3C(NC(C=Cc4scc(C)n4)=O)CC(C3)C2)=O)cccc2c1CCO2 60430,c1(C(=O)NC(CCN(C(CC2(C=C)CCCCC2)=O)C)C)coc(S(N)(=O)=O)c1 60431,C1(CC)CCCCCCN1C(C1CCN1CC)=O.C12OCCC1NC2=O 60432,c1(C(N(CC(CNC(C(C)C#N)=O)O)C)=O)nn(C)c2ccccc2c1=O 60433,c1(CNC(C2CC(F)CN(C(c3ccc(I)c(Cl)c3)=O)C2)=O)cccc(F)c1Cl 60434,C(C(=O)N1CCCC(CN(C(=O)CCOCCN(C)C)C)C1)(C(C)C)OC 60435,CC(C)CCC(=O)NCC(=O)NC1CCC(NC(c2nc(C3CC3)cs2)=O)C1 60436,CC1(CNC(=O)CCC(N)=O)CCN(C(=O)C(c2ccccc2)O)C1 60437,c1(C(N2CCCC(NC(C(C)OCCC=C)=O)C2CC)=O)cnc2n1CCCC2 60438,n1(CC)nc(C(=O)NC2CCN(C(c3cnc(N(C)C)s3)=O)C2C)c(C)n1 60439,N1(C(c2cnc(CCC)s2)=O)CC(C)(C)CCC1CNC(C1CCCN1N=O)=O 60440,C(=O)(CS(C)(=O)=O)NCC1CC(CC(=O)NC(c2ccon2)(C)C)C1 60441,N1(C(C(C)(C2CCC2)NC(=O)Cc2ccsc2)=O)CC2CC(O)CC2C1 60442,CN1N=C(CC(=O)NC2(C)CCN(Cc3ccncc3Cl)C2)CC1=O 60443,c1(CC)ccc(C(=O)NC2(CNC(c3ccoc3Br)=O)CCOC2)s1 60444,C1(C(=O)NC2(C)CN(C(C(COC)(F)F)=O)C2)CC2(CCC2OC)C1 60445,C1(NC(c2[nH]cc(CC)n2)=O)CCCN(C(c2cc[nH]c2CC)=O)C1C 60446,CCCC(C)C(C)NCC1CC1C(=O)OC(C)(C)C 60447,C1(NC(C(CCC)CNC(=O)CCCN(C)C(C)=O)=O)C2CCCCCCC12 60448,Nc1cnc(C(=O)NC2CCC2NC(c2cccn2C2CCCC2)=O)cn1 60449,c1(C(N2CC3CC2C3C(N2CCC2(CO)CO)=O)=O)ccc2[nH]nc(Cl)c2c1 60450,c1(C(=O)NCCOC(CNC(c2cnc(CCC)s2)=O)(C)C)cnc(N)c(Cl)c1 60451,C(C1C(C(=O)NCCC2(NC(c3ccc(CSC)cc3)=O)CC2)C1(C)C)=C(C)C 60452,c1(C(C(=O)NCCC(=C)CNC(c2ccnc(OC)c2)=O)O)ccc(Cl)c(Cl)c1 60453,N1(C(c2cnc(C(C)OCC)s2)=O)CCC(NC(c2ccc(C)o2)=O)CC1C 60454,N1(C(C2C(=C)C2)=O)CC(NC(=O)Cc2cccc(C(N)=O)c2)CC1(C)C 60455,C(=O)(CC(C(F)(F)F)n1ccnc1)NCCC(C)NC(c1ncc(F)cn1)=O 60456,C=CCC(CNC(c1ccncc1Cl)=O)C(=O)N1CCC(C(F)F)CC1 60457,c1(C(=O)NCCn2ccc(C(=O)NCCc3ncn(C)c3)c2)ncc(F)cc1F 60458,Cc1cn2c(n1)C(C(=O)NCC(C1CC1)NC(=O)C(C)(C)N(C)C)CCC2 60459,c1(C(=O)NC2C(CC(=O)NC(CC#C)CC)C(O)C2)nccnc1C 60460,c1(CN(C(C(C)NS(C)(=O)=O)=O)CCOCCO)cnn2ccncc12 60461,c1ccc2c(N3CCC(OCCC4CCCCN4)CC3)nsc2c1 60462,C(c1ccsc1)=CC(=O)NCC(C1CCOC1)NC(C1CC(=C2CCC2)C1)=O 60463,CC=C=CCCN=c1nc(N2CCN(C)CC(C)C2)c2ncccc2[nH]1 60464,c1(C(=O)NC2C(CNC(C3CC(=C)C3)=O)C2)cc2c(N(C)C)cccc2s1 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60482,S(=O)(=O)(c1ccc(Br)cc1C(=O)O)NCC(c1cc(C)cc(C)c1)O 60483,CC(C)(C)C(=O)C(=O)NCC1CCC(CC(=O)NCCCCCCF)CC1 60484,C1(NC(=O)Nc2cc(C)c(I)cc2)(CO)CC(O)C12CCC2 60485,C1(CCNC(C2(C)CC(F)C2)=O)CCCN(CCC(=O)NCc2ccccc2)C1 60486,c1(C(=O)NC2(CC(=O)Nc3ccc(C)cc3O)CCC2)ccc2ccn(C)c2c1 60487,C1(C(=O)NCC(C(F)(F)F)OC)CNC2(CC2)CO1 60488,c1(CC)ncc(C(=O)NC(C)CCNC(c2sc(=N)[nH]c2CC)=O)cn1 60489,N1(C(C(C)O)=O)CCc2[nH]nc(CNC(=O)CCC3CCOC3)c2C1 60490,S(=O)(=O)(c1csc2ccccc12)NC1CN(C(c2nc(Cl)ccc2F)=O)CC1O 60491,C(=O)(CCC(C)C)NCC(CCOC)NC(=O)CCC1CCCCO1 60492,CC(C)C(CCC(=O)N1CC2CC3CC2C1C3)NC(C1OCCC1(C)C)=O 60493,C(CS(=O)(=O)CC(=O)NCC1CCN1C(=O)CCCC(C)O)OC 60494,CC1(Cc2ccc(Cl)c(Cl)c2)CCCN1N1CCCC2(CC1)CC2(F)F 60495,N1(C(c2ccc(OC(C)C)nn2)=O)CCC(NC(c2coc(Br)n2)=O)C(O)C1 60496,C12(NC(C(=O)NCC3CC3)=O)CCC(CC1)N(C(c1ccncc1)=O)C2 60497,C(CC(=O)NCCc1nccs1)N(C(C)C)C(C1CC(=C2CC2)C1)=O 60498,CC(C(=O)N(CCNC(=O)CC1CN(C)C1)CCOCCO)c1ccsc1 60499,N1(C(C(C=C)OC)=O)CC(C2CCCN(C(=O)CC3CC4CC4C3)C2)C1 60500,C1(CC(c2nnnn2CCCC2CC2)NC(C)C(=O)NO)CCC(C)(C)CC1 60501,c1(C(=O)OCC)cc(NC(C2(C)CCCN2C(c2ncco2)=O)=O)ncn1 60502,C1(CN(C(=O)CN2CCCC2CO)C)CCCN(C(c2cccc(O)c2)=O)C1 60503,N1(C(C(CC(C)C)ONC(=O)CC(C)c2ccco2)=O)CC2(C1)CC(C)(C)C2 60504,c1(C(N2C(CC(=O)NCCc3ccccc3Cl)COCC2)=O)cccc(F)c1Cl 60505,n1(CC(=O)Nc2cccc(NC(C3CCC(=O)NC3=O)=O)c2)ncc2ccccc12 60506,CC1(C(=O)NCC2C=CCN2C(=O)CCc2ccc[nH]2)CC(F)C1 60507,N1(C(C2C(C)(CC)C2)=O)CCOC(CNC(=O)CCCCN2CCOCC2)C1 60508,C(=O)(NN1CCN(Cc2ccccc2)CC1)c1c(-c2c(C)n[nH]c2)csc1 60509,N1(C(c2cc(-c3ccc(C)o3)[nH]n2)=O)CCC(NC(c2ccn(C)n2)=O)CC1C 60510,c1(OC)csc(C(=O)NC(C)CC(C)NC(=O)CC2(OC)CCC2)c1 60511,c1(C(N2CCC(C)C2CNC(=O)CC2(C)CC2(Cl)Cl)=O)cc[nH]c2nccc1-2 60512,C1(C(N(C2CCC2)Cc2c(C)nc[nH]2)=O)CCCC(=O)N1C.C12(O)CC(C1)CS2 60513,c1(C(N(CCN(C(c2cccc(OC)c2)=O)C(C)C)C)=O)ccc2c[nH]nc2n1 60514,N1(C(c2nc(N(C)C)oc2)=O)CCOC2(CCN(C(C3CCCC(F)C3)=O)C2)C1 60515,Cc1c(C(=O)NC2C(C(=O)NC(C)CCC(C)C)C2(C)C)cccc1F 60516,c1(C(=O)NC2C3C(C)N(C(CC(C(C)C)O)=O)C2C3)ccn2ccnc2c1 60517,C1(C(=O)NCCC2(CNC(C(CSC)O)=O)CC2)CC(=O)N(c2nccs2)C1 60518,c1(NC(C(c2cn(C)nn2)NC(CSCC=C)=O)=O)ccccc1F 60519,c1(C(=O)NC(CNC(CCC(C)C)=O)C2CCC2)c(C)oc2ncnc(O)c12 60520,C1(NC(C(SC)SC)=O)C2CC(NC(C3CCN(C)C3C)=O)CC12 60521,c1(C(=O)NC(CCC)CNC(=O)C(C)=C(C)C)cc(Cl)nn1C 60522,C(=O)(C1CC(=O)Nc2ncccc21)NC(C)(C)CCCNC(c1ccc(F)s1)=O 60523,c1(NC(CC)C(=O)NCC(C)(C)NC(=O)Cc2cncn2CC)cccc(C)c1 60524,c1(C(=O)NCCN(CCCCCC)C(c2ccsn2)=O)ncc(N)cc1Cl 60525,c1(C(CN(C2CCN(C(=O)CCC3CC(F)(F)C3)C2)C)O)cc(F)ccc1F 60526,C1(CNC(C2CCC(C)(C)C2)=O)CC(F)(F)CN1C(=O)CCCN1CCCC1 60527,C(=O)(C(C(C)(C)C)N1CCNC1=O)NCC(C)CNC(=O)Cc1ccco1 60528,C(=O)(C(CC(C)C)ONC(C1COCCN1C)=O)N(CCOC)CC 60529,C1(C(=O)Nc2cccc(C)c2C#N)C2CCCC1CN(C(c1c(C)cc[nH]1)=O)C2 60530,Cc1cc(C(=O)NC2(CCNC(C3CC(OC(F)(F)F)C3)=O)CC2)c(C)c(C)c1 60531,c1(C(C)(C)C)cccc(C#CCN(CCO)Cc2cc(Cl)c(Br)cc2F)c1 60532,C1(NC(CC2(OC)CCC2)=O)CCN(CCCOC(C)=O)C1.C12CN(C1)C(=O)C2 60533,C1(C(N(C)CC2(NC(C=CCCC=C(C)C)=O)CC2)=O)Cc2cccnc2C1 60534,CCC(CNC(c1conc1CNC(C1CNC(=O)N1)=O)=O)CC(C)C 60535,C1(C(N(C(C)C)CCNC(C2(c3ccc(O)cc3)CC2)=O)=O)CN(C)CCO1 60536,CCCC(C(=O)NC1CC1CNC(=O)Cn1cc(Cl)cn1)c1ccc(Cl)cc1 60537,CC(=O)CCCC(=O)N1CCN(C(C23CCCCC2C3)=O)CC1C 60538,c1(CNC(=O)C(F)(F)F)ccc(F)c(-c2c[nH]c(=NCc3ncccc3Br)s2)c1 60539,N1(CCOC)CCCC(C(C)NC(=O)CCc2ccccc2Cl)C1 60540,c1(CC)nocc1C(=O)NC(c1cnn(C)c1)C(=O)N(C)CCOCCOC 60541,c1(CC(=O)NC2C(NC(C3C=CCCC3)=O)CCC2)cccnc1C(F)(F)F 60542,c1(C(c2nnnn2C)NCCc2nc(C(=O)OCC)sc2)c[nH]c2cccc(F)c12 60543,c1(C(N2C(CC(=O)OC)CC2)=O)cc(Br)ccc1C 60544,C1(CCCC)CN(C(c2n[nH]c(C)c2Br)=O)CCN1C(=O)CC(C)F 60545,C=C(F)C1(CC(N2CCC(CNC(C3(OC)CCOC3)=O)(OC)C2)=O)CCC1 60546,S(=O)(=O)(c1ccc(F)cc1F)C(c1cc(C(C)C)no1)=O.C1(N)CC2CC1CN2 60547,c1(C(C)OCC)noc(CN(C)C(C2(C)CCCS2)=O)n1 60548,c1(C(=O)NC2CC(NC(Cc3nc(C)sc3)=O)C2)ncnc2sccc12 60549,C1(C(=O)NC2CCC(NC(c3nc(Br)c[nH]3)=O)C2)CCC2(CCC2)C1 60550,CCC(C)C(C)(O)CNC(C1CCCC1CNC(c1cncc(O)c1)=O)=O 60551,CC(C)C(C)(CNC(c1ccc(-n2ccnc2O)cc1)=O)NC(=O)C1=NOCC1 60552,N1(C(C2CCCN(C(c3c(CC)nns3)=O)C2)=O)CCC2(CCCC2)C1 60553,c1(C(N(CC(C)(C)NC(C2=CCCC2C)=O)C)=O)cnc2ncnn2n1 60554,C(CN=c1c(C#N)c[nH]c2ccc(C)cc12)N(C(C1CCC(C)C1)=O)CC 60555,O=S(=O)(c1cnc(NCC(C(F)(F)F)SC)c(Cl)c1)NCC1CC2CCCC(C1)C2 60556,c1(C(=O)NC2CCC(NC(CC(CC)OC)=O)CC2)ccc2c(c1)CCN(C)C2 60557,c1(C(=O)NC2(C)CCN(C(c3c(N(C)C)cccn3)=O)C2)ccc(P(C)(C)=O)s1 60558,C1(CC)CN(Cc2ccccc2N(C)C)CCN1C(=O)Cc1ccsc1 60559,C1(C(=O)NCC(C2CC2)SC)CC2CN(C(=O)Cn3nnc(C)n3)CC2C1 60560,c1(OC)ccc(C(=O)NCC(CO)NC(=O)C(c2ccccc2)OC)cc1 60561,CCCC(C)(C)CC(=O)NC(CCC(=O)N1CCC1C(N)=O)C(C)C 60562,C1(CC)(CNC(C2(NC(c3ccn(C4CC4)n3)=O)CC(O)C2)=O)CCOC1 60563,c1(SC)cc(C)nc(N2CC(NC(C3(C4CC4)CC3)=O)C(C#N)C2)n1 60564,Cc1ccc(C(=O)NC2(CS(N)(=O)=O)CC2)nc1C 60565,C(=O)(C(C)(CSC)NC(=O)C=Cc1ccoc1)NC(C#C)C 60566,C1(C(N2CCCC(C(=O)OC)C2)=O)CC(C)(C)CN1C(=O)CC(C)F 60567,C(C(C)(C)CNC(c1ncoc1C1CCC1)=O)N(C)C(c1coc(Br)n1)=O 60568,CC1C2CCCCC2CN1C(=O)C(CC1CC1)NC(C1CCC(=O)O1)=O 60569,c1(CSCCC(=O)NCCC2CCN(C(CC(=O)NCC)=O)C2)ccc(F)cc1 60570,N1(C(c2ccc(C#C)cc2OC)=O)CCC2C(CCCN2C(=O)CC(C)(C)C)C1 60571,C=CC1(C(=O)NCCCc2ncn(C)n2)CCN(C(=O)CCc2cccs2)C1 60572,CC1(C#CC(=O)NC2CC3CCC2N3C(c2cc(Cl)c(Cl)s2)=O)CC1 60573,C1(C(=O)NC2CCN(C(C)=O)CC2)CCC2(CN(C(=O)C(O)C(C)C)C2)O1 60574,C1(NC(C2(C)CNC(=O)C2)=O)CN(C(=O)CN2CC(=O)NC2=O)CC1C1CC1 60575,c1(C(=O)NC(C2CCN(C(=O)C(C)(C)C(=O)NC)C2)CC)nccc(Cl)c1C 60576,CCC(C)CC(C)C(=O)NCC(C)=CC(=O)Nc1cc(CO)cc(C)c1 60577,CC(CC(=O)NCCCC(=O)NC(N)=O)N(C)C(C1CCS1(=O)=O)=O 60578,C=CCC(CC(=O)N1CCC(COC)CC1)NC(=O)C(CC=C)OC 60579,C1(F)(CNC(=O)CC(F)F)CCCN(C(=O)Cc2ccon2)CC1 60580,CC(CC(=O)NC1(CF)CCN(C(=O)C(C)OCCOCCO)C1)C(F)(F)F 60581,C(CCCCC(=O)NCC1CCCCN1C(=O)CCC1CCCC1)N(C)C 60582,c1(C(=O)NCC2CCN2S(=O)(=O)C2CC2)nc(C(F)(F)F)ccc1Cl 60583,C1(C(=O)NCCCC(C)NC(C2CCC3(CC3)C2)=O)C2CC3C(C2)C13 60584,CC1(C)CCCN(C(C2CS(=O)(=O)C2)=O)C1CNC(c1cnc2ccsc2c1)=O 60585,C1(NC(C(C=C=C)C)=O)CCCCN(C(c2cnc(OC)s2)=O)C1 60586,CC1(NC(=O)CC2CCCC23CC3)CCN(C(=O)Cn2nnc(=N)[nH]2)CC1 60587,CC#CCCCC(C)N(c1ccc(C(C)(C)C)cc1)CCC#N 60588,c1(OC)ccc(F)c(C(=O)NCC(C)(C)CN(C)C(C2CCCC2(C)C)=O)c1N 60589,C(C(C)C(C)C(=O)N1CCCC1CN(C(=O)CCNC(c1ccco1)=O)C)OC 60590,CC1CC(ONC(N2CCCC2Cc2ccccc2)=O)CCO1 60591,C12(CNC(C3CC3(F)F)=O)CCCC1N(C(c1ncnc3sccc13)=O)CCC2 60592,C1(CNC(c2cncc(OC)c2)=O)CCN(C(=O)CC(C)N(C)C)C12CCC2 60593,C1(NC(CC2(OC)CCCCC2)=O)CC(C)CN(C(=O)CCc2csc(=N)[nH]2)C1 60594,C1(CCC)(NC(=O)CCc2cnoc2)CCN(C(c2ccc([N+](=O)[O-])s2)=O)CC1 60595,C1(C(=O)NCCC2CCN(C(C(c3n(C)ccn3)(F)F)=O)C2)CCC(F)(F)CC1 60596,N1(C(c2cn(CCC=C)nn2)=O)CCN(CC(C)NC(c2n[nH]cc2Cl)=O)CC1 60597,CCC(C)(CN(C(=O)CN1CC2CC2C1)CCOC)C(=O)N1OC2CCC1CC2 60598,C#CC1CCN(C(C2COCCN2C(=O)C(C)=C2CCCC2)=O)CC1 60599,CC1(C(=O)NC2CN(C(c3cccc[n+]3[O-])=O)CC2CO)CCC(O)CC1 60600,c1(C(=O)Nc2nc(C)c(-c3nn[nH]n3)s2)n[nH]c2cc(Br)ccc12 60601,c1(CNC(C2CCN(c3ncc(C#N)nc3)CC2)=O)nnn2c1COCC2 60602,C12(NC(CC(COC)NC(=O)Cn3nc(C)nc3C)=O)CCC(C1)OC2C 60603,C1(NC(CNC(CC)=O)=O)(CC)CCN(C(C2CC2Cl)=O)CC1 60604,C=Cc1cccc(CN2CCCC(NC(=O)CCc3ccccc3)C2)c1 60605,C1(NC(C(C)(CO)OC)=O)CN(C(c2cc(C)cc(Br)c2)=O)CC1N=[N+]=[N-] 60606,c1(C(C(=O)NC(C(=O)OC)C)N(C(C)CCO)C)ccc(OC)c(Br)c1 60607,CCCCC(O)C(C)C(=O)NCC(C)=CC(=O)NCC(O)CCC1CC1 60608,c1(C(N(CCC)CCNC(C2CC2C(C)(F)F)=O)=O)cnc(C(C)C)nc1 60609,CC(CC(C)(C)C)C(=O)NCC(C)(CO)NC(=O)CCCn1cncn1 60610,c1(C(=O)NCC2N(C(C(C)=C(C)C)=O)CC(F)C2)cccc(=S)n1O 60611,c1(OC)ccccc1C(N1CCCC(CCNC(=O)CC(O)CN(C)C)C1)=O 60612,Nc1cccnc1S(=O)(=O)NC1CC(=O)NC1=O 60613,c1(C(=O)NC(C2N(C(CSCCC)=O)CCC2)C)cccc2nc(COC)[nH]c12 60614,c1(C(N2CC(C)C(NC(=O)C(C)(C)N3CCCC3)C2)=O)cc(N)c(Br)c(F)c1 60615,N1(C(N(C2CCCN(C)C2)C(C)COC2CCCCC2)=O)CC2CCC(CO)(C2)C1 60616,C=C(C)C1OCCCC1C(N1CCC2(C1)CN(C(c1cc(O)ncn1)=O)C2)=O 60617,C1(NC(C=C(C)c2ccsc2)=O)CC2CCC(C1)N2C(=O)C(C)S(C)(=O)=O 60618,CN1CCNC(=O)C12CCCN(CC(c1cnc3ccc(Cl)nn13)=O)C2 60619,C1(C(=O)NCC2(CO)CCCC2)CC2(CCC2)CN1C(c1ccnc(O)c1F)=O 60620,C(c1ccc(Cl)cc1)=CC(=O)N(C)CC1(NC(=O)C(C)(O)C2CCOC2)CC1 60621,C1(NC(=O)CC2CC3C=CC2C3)CC2CC1N(C(C1CCCCC1)=O)C2 60622,c1(C(N2C(C(N3CC(CC)C3)=O)CNC(=O)C2)=O)ccc2[nH]ccc2n1 60623,C1(OC)CCC2(C(=O)NCC(C)C(=O)NCC(c3cnc[nH]3)C)CC12 60624,Cc1cc(Br)cnc1C(N1CCC(NC(=O)CCN2CCC2)C1C1CC1)=O 60625,C(CN=c1nc2c(ncn2C)c(NC2CCN(C)C(C)C2)[nH]1)OCCOCCC 60626,c1(C(=O)NCC(CC(F)(F)F)NC(=O)C(O)C2CCC2)cc2ccc(F)cc2o1 60627,C1(NC(c2c(CC)nc[nH]2)=O)CC2(CCN(C(=O)C(C)CCCOC)C2)C1 60628,C(CCC(O)C(=O)NC1CCOC(C)(C)C1)NC(C(CCC)NC(C)=O)=O 60629,N1(C(CCCc2onc(C)n2)=O)CCC2(NC(c3cnc(C(C)C)[nH]3)=O)CC2C1 60630,N1(C(CCCCN(C)C)=O)CC2CCN(C(c3snc(Cl)c3Cl)=O)CC2C1 60631,Cc1cnc(C)c(C(=O)NCC(C)CNC(=O)CSc2ccc(F)cc2F)c1 60632,c1(C(=O)NC2C(NC(C(CC)(C)C#N)=O)CC2)cc2c(cc1F)OCC(=O)N2 60633,N1(C(CC)=O)CCCC(C(=O)NC(C)(CNC(=O)C2=COCC2)C(C)C)C1 60634,c1(CSC)cc(C)c(C(N2CCC(C(C)(C)C)(CNC(C3(O)CC3)=O)C2)=O)s1 60635,C(=O)(C(C)C(C)(C)C)NCc1cc(C(=O)NCC(C#C)C(C)C)sc1 60636,c1(C(N(C)CCOCC2(O)CCOC2)=O)ncc(C(C)(C)O)cn1 60637,c1(OC)cnc(Cl)nc1N1CCCC(C(C)NC(c2cnncc2O)=O)C1 60638,C1(NC(c2n(C)cnc2)=O)COC2(CCCN(C(C3(CO)CCOCC3)=O)C2)C1 60639,c1(-c2cc(CCN(C)C)on2)nc(C2CCCCC2)nn1CCS(C)(=O)=O 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60674,N1(C(C2CC(C)C2)=O)CC(NC(=O)Cn2nnc3ccccc23)C2(CCCC2)C1 60675,C(c1ccc(Cl)cc1F)=CC(=O)NC1CC(F)(CNC(C23CC(C)C2C3)=O)C1 60676,N1(C(CC2(C)CCCC2)=O)CC(CNC(c2cccc(F)c2Cl)=O)CC12CCC2 60677,N1(C(C2(CC)CCC2)=O)CCCC1C=CC(=O)NCC1(O)CCN(C)C1 60678,c1(CC(N2CC(NC(C=CC(C)(C)C)=O)C3C2C3)=O)ccc2c(c1)OCO2 60679,c1(C(=O)NCCC2COCCN2C(=O)CCOCC2CC2)nccc2n[nH]cc12 60680,c1(CC(=O)NCC2(O)CC(NC(c3cnc(OC)s3)=O)C2)cc(C)ccc1OC 60681,N1(C(C(CCC)C)=O)CC2(C1)CN(C(C1(C)CCCC1)=O)CC2CO 60682,C1(NC(CCNC(=O)NC)=O)CCC(O)CN(C(c2cn(C)c(O)n2)=O)C1 60683,N1(C(CC2CC(=C)C2)=O)CCN(C(c2ccc(N)cc2OCC)=O)CC(C)(C)C1 60684,Cc1nc(O)c2c(n1)CCN(C(c1ccsc1S(C)(=O)=O)=O)C2 60685,N1(C(C(N2CCCCC2)C)=O)CCOC(CCCNC(=O)CP(C)(C)=O)C1 60686,C(=O)(C(=O)N=S(C)(C)=O)NC1C(C)CN(C(c2ccc([N+](=O)[O-])s2)=O)CC1 60687,C1(O)(C(N(CCC)C)=O)CCN(C(c2nnc(C)s2)=O)CC1 60688,c1(C(N2C(CCCNC(CSC)=O)CCC2)=O)ccc(F)cc1N 60689,CN1CC=C(CC(=O)NC(C)(CNC(C23CCCC2OCC3)=O)C2CCC2)CC1 60690,c1(C(N(CC2CCN(C(C=CC(=O)OCC)=O)C2)CC)=O)cn2c(n1)SCC2 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60759,CC1(C)CC(NC(C2SCCS2)=O)CN1C(C1CC1C1CC1)=O 60760,CC1CCS(=N)(=O)CCN1C(=O)C(C(C)(C)C)n1cc(C2CCC2)nn1 60761,C(C)(CNC(c1ncccc1Cl)=O)(CC(C)C)NC(C(CC)OC)=O 60762,C1(NC(C=CC)=O)COC2C(NC(c3c(Cl)ccc(F)c3F)=O)COC12 60763,N1(C(C2CC(CCC)C2)=O)CCC(C(=O)NC2(CC(C)(C)C)CC2)C1C 60764,N1(C(CCC)=O)CC(NC(=O)C(O)Cc2cn(C)cn2)CC12CCOCC2 60765,C1(CN(C(=O)CCc2ccnc(Cl)c2)CC)CCN(C(=O)C(C)C2CCC2)CC1 60766,c1(C(CNC(C2(COC)CCCC2)=O)NC(=O)C(O)C2CCC2)ccccc1F 60767,N1(C(C(c2cccs2)NC(Cc2c(C)nccc2)=O)=O)CC(=O)N2CCCC2C1 60768,C1(C(N2CCN(C(CC)=O)CC2C)=O)CN2CCCN1CC2 60769,N1(C(C=CSC)=O)CC(NC(c2ccc(F)c(F)c2N)=O)C(C2CC2)C1 60770,N1(C(c2cn(CC)nc2)=O)CCCC(N(C)C(c2cc(CO)[nH]n2)=O)CC1 60771,n1(CCCC)nnnc1C(c1ccccn1)NCC(C)(C)SC 60772,CC(CCC(C)(C)C)NC(=O)CN(C(c1cc(F)cnc1O)=O)C1CC1 60773,c1(CN(CC(N2CC(N(C)C(=O)NC(C)(C)C)C2)=O)C)ccc(C#N)cc1F 60774,c1(N(CCOCC=C)C)nc(=NC(C)c2ccc(F)c(Cl)c2)[nH]c2c1CSC2 60775,C1(C(=O)NC23C(CN(C(C(C)(C)OC(C)C)=O)C2)C3)CCOC(=O)CC1 60776,O=S1CCC(NCC(=O)NC2CCN(c3ccccc3)CC2)=N1 60777,c1(C(N(C)CC2CN(C(=O)CC(C)(O)C3CC3)CCO2)=O)cc(O)nc(O)n1 60778,C1(CCC2N(C(c3c(OC)ocn3)=O)CCC2)CCCCN1C(C)=O 60779,Cc1ccc(C=CC(=O)NCC2(CNC(c3occc3C)=O)CCC2)cn1 60780,N1(C(C2CC=C(C)CC2)=O)CCCC2(NC(c3ccc(Cl)nc3Cl)=O)CC2C1 60781,Cc1ccc(OCCCC(=O)N(C)CCNC(=O)C(C)N2CC(C)C2)cc1 60782,c1(C(=O)NCCN(C(=O)CCC(C)OCC)CCC)c[nH]c2c(CC)cccc12 60783,c1(OCCC(=O)NC2CCC(CCNC(C=NOC)=O)C2)ccc(OC)cc1 60784,CC1(C)CC(CNc2cc(N3CCC(Cc4ccncc4)CC3)ncn2)CO1 60785,N1(CC(=O)NCC(CCCC)NC(=O)Cc2occc2C)C(=O)CN(C)C1=O 60786,CCCCCCN(C(=O)Cn1cccn1)CCN(C(C1CCCC1C)=O)CC 60787,Cc1cc(NC(c2ccc(S(C)(=O)=O)o2)c2nnnn2C(C)(C)C)cc(C)c1F 60788,c1(C(=O)NCCC2(NC(C3C(C(=O)OC)C3)=O)CC2)sc(Cl)c(Cl)c1C 60789,C1(C(=O)NC2C(CNC(C(c3ccc(C)cc3)=O)=O)CC2)CC12CCSCC2 60790,c1(C(=O)NC2CC3CC(NC(C(F)=CC)=O)C3C2)c[nH]c2ccc(Cl)cc12 60791,c1(C(=O)NCC#CCNC(CCC2OCC(C)(C)C2)=O)cc(Cl)ccc1Cl 60792,c1(C(=O)NCC2CCN2C(c2cnco2)=O)cnn(CC2CCCCO2)c1 60793,C(CCC(=O)NC1(C(=O)NCC(c2cccs2)C)CCC1)NC(C)=O 60794,C(=O)(C#CC1(C)CC1)N(C)CC1CCCN1C(c1cn(C)c(C(F)F)n1)=O 60795,CCCCCC(C)CC(=O)N1CCC(C)C(CNC(c2cc(SC)oc2C)=O)C1 60796,Cc1cc(C(N2CCCCC2CC(=O)NCc2noc(C3CC3)n2)=O)sc1C 60797,c1(C(C)(C(=O)NC2CC(F)(F)C2)N(C2CC2)Cc2ccccc2)ccc(Br)cn1 60798,c1(CCCC(=O)NC2C(OC)CN(C(c3cnoc3C)=O)C2)ccc(F)c(F)c1 60799,c1(C(N2CC(NC(=O)CCC3CC3)CC(C)C2)=O)ccc2nc3n(c2c1)CCC3 60800,c1(CNC(c2n(CC)nc(C)c2)=O)ccc(CNC(=O)C(C)NC(C)=O)cc1F 60801,CC1=C(C)CC(C(=O)NCC2CCC(C(N3CCCC(CN=[N+]=[N-])C3)=O)C2)CC1 60802,C1(CC(N2CCC(CC(=O)N(CCC(=O)OC)C)C2)=O)CCC(=O)N1C 60803,C1(C)(NC(C2N(C(C(C)C)=O)CCC2)=O)CCS(=O)(=O)C1 60804,CCC(F)(F)CC(=O)N1CCCC(C2CCCCN2C(C23CSC(C2)C3)=O)C1 60805,C1(NC(c2ncn(CC)c2)=O)CCCC2CN(C(c3c(Cl)cccc3Cl)=O)CC12 60806,N1(C(C2(C)CC(C)C2)=O)CCC(NC(=O)C=CSc2nc[nH]n2)C(O)C1 60807,CC1(C)C(CC(N2CCOC3(CC3)C2)=O)CCN1C(=O)Cn1cnnc1 60808,C1(CC)CN(C(c2cnc(Cl)cc2I)=O)CCN1Cc1ccnc(OC)c1 60809,c1(C(N(C)CC2CCCN(C(C3CCC3(F)F)=O)C2)=O)cc2nc[nH]c2cc1F 60810,CC1(CNC(C2C=CCN(C(c3nc(Cl)cs3)=O)C2)=O)CC2CCC1C2 60811,N1(C(CCc2nc(C)sc2)=O)CCc2c(CNC(=O)C=CC(C)C)cccc2C1 60812,c1(C(C)(C)C#N)cccc(C(=O)NCC(F)CNC(=O)CC2C=CS(=O)(=O)C2)c1 60813,N1(C(c2c(C)nn[nH]2)=O)CC=C(C(=O)NCC2CCN(C3CC3)C2)C1 60814,N1(C(C2CC23CC3)=O)CCN(C(=O)C(F)CC2CC2)C2(CC2)C1 60815,c1(CC(=O)NC2CCN(C(C=C(C)C3CC3)=O)C2C)cc(C(F)(F)F)c(O)nn1 60816,C(CCCCC(=O)NCC1(F)CCC(NC(=O)C=Cc2ccco2)C1)=CC 60817,N1(c2nnc(OCC)s2)CCC(C)C(NC(c2cnn(C)c2C)=O)C1C 60818,N1(C(C(C)CC2CC2)=O)CCOC2(C1)CN(C(=O)C(c1ccc(Cl)cc1)CO)C2 60819,Cn1cc2c(n1)CCCC2C(=O)N1CCCCC1CNC(=O)CC#N 60820,C(N=c1[nH]c2c(c(=NC(C)c3c[nH]nc3C)[nH]1)CCC2)C1(CSC)CCOCC1 60821,C1(C(C)CO)CCCCN1C(c1coc(CNC(c2ccc(C(F)F)o2)=O)c1)=O 60822,C1(NC(C(C)Cc2ccccn2)=O)CC2CC1N(C(=O)Cc1csnn1)C2 60823,N1(C(CSCC=C)=O)CC2CCCCC2(NC(=O)Cc2cccc(O)c2)C1 60824,CCCC(C(O)C(=O)NC1CCN(C2CC2)C1)NC(C1(n2cccc2)CC1)=O 60825,c1(C(C)Cc2nc(-c3cccc(F)n3)no2)ccc(S(C)(=O)=O)cc1 60826,C(C1c2ccccc2CN1C(C1C2(CC2)C12CC2)=O)NC(C(C)OCC(C)C)=O 60827,N(C1CCCn2ncnc21)C(C(C)N(C(=O)CC(C)C(F)(F)F)CCC)=O 60828,Cc1nc(C(=O)NC2(CNC(C3CCCN3C3CCCCC3)=O)CC2)cc(O)n1 60829,C=CCCCC(C(=O)N1CC(=CC)C1)NC(C1C2CCCCC12)=O 60830,C1(NC(c2c(CC)non2)=O)CCCC12CN(c1nc(Cl)nc(C)c1F)C2 60831,C1(C)(C(=O)NC(CC)CN(C(c2cc(-c3ccoc3)on2)=O)CC)C=CCCC1 60832,N1(C(C(=O)NC(C)C)=O)CCC2(CCN(C(c3cccnc3NC(C)C)=O)C2)C1 60833,c1(C(=O)Nc2ncc(Br)cc2I)cc2c(s1)CCN(Cc1cc(Cl)cc(I)c1)C2 60834,CON1CCC(CC(=O)NCCOCCN(C)C(C2(C)CCCS2(=O)=O)=O)CC1 60835,C1(N(C(C(C)=C2CC2)=O)C)CC2CCC(C1)N2C(=O)COc1ccsn1 60836,C1(CC(C)NC(c2ccc(N)cn2)=O)CCN(C(=O)Cc2cncs2)CC1 60837,CC(C)(C)C(=O)C(=O)N1CC2(CCC2NC(=O)CNC(C2CCC2)=O)C1 60838,Cc1c(C(F)(F)F)cccc1S(=O)(=O)NCCCSC(C)C 60839,c1(CC)ccccc1CN(C(C)CNC(=O)C(COC)OC)C 60840,c1(OC)cccc(-c2nc(CC(=O)Nc3c[nH]nc3C#N)cs2)c1OC 60841,c1(CC(N2CC3C(C(N4CCC(CC)C4)=O)(C3)C2)=O)cccc(C#N)c1 60842,N1(C(C2CCN2CC2CCC(F)C2)=O)CCCCC1CO 60843,N1(C(C2CCC(OC(C)C)CC2)=O)CCCN(C(c2cccc(=O)o2)=O)CCC1 60844,CCCCC(O)C(=O)N(C1CCCCN(C(=O)CC2(n3cccn3)CC2)C1)C1CC1 60845,C1(CN(CCC)CCNC(C2CC3CCC2C3)=O)CCC(F)(F)C1 60846,N(C(=NCCCF)N1CCC2C(C1)NC(=O)N2C)Cc1c(C)nn(C)c1C 60847,C1(CC)(OC)CN(C(=O)C(C2(C)CC2)NC(c2csc(C3CC3)n2)=O)C1 60848,c1(C(CC)=O)ccc(C(=O)NCC2(O)CN(C(=O)CC(C)NC(N)=O)C2)cc1 60849,CC1CN(C(C2CC(C)(F)C2)=O)CCC1NC(c1cc(O)cs1)=O.C1CC1 60850,C=C(C)CC(C)C(=O)NCC(C)(C)NC(c1ccsc1C)=O 60851,c1(CC)ccc(C(=O)N(C2CN(C(=O)C#CC3(C)CC3)CC2(C)C)C)c(O)c1 60852,N1(CC(=O)N(C(C)CN(C)C(c2cc(O)ccc2F)=O)C)Cc2ccccc2C1 60853,N1(C(Cc2ccc(C)cc2)=O)CCC(O)C(N(C(=O)C(O)C2CCC2)C)C1 60854,N1(Cc2ccc(C(=O)NCCC(C)OC)o2)CC2CCC(NC(C)=O)CC2C1 60855,N1(C(C2CN(C(N)=O)C2)=O)CC2CC(NC(=O)CCC3CC3(F)F)CC(C2)C1 60856,Cc1ccc(CCC(N2CC(O)(CCNC(C3CC3(C)C(F)F)=O)C2)=O)o1 60857,C1(c2c(C(=O)NC3C(C)C3C)c[nH]n2)CCCCN1C(c1cnnc(O)c1)=O 60858,c1(C(=O)NC(CCNC(CC2(COC)CC2)=O)C(C)C)ncc(C)cc1F 60859,CC1C(NC(c2c[nH]cc(F)c2=O)=O)CCCN1C(c1ccccc1F)=O 60860,C1(CCC)(NC(=O)Cc2cn(C)nc2Cl)CCCN(C(=O)C2=C(C)CCC2)C1 60861,c1(-c2onc(C(c3ccccc3Cl)(C)C)n2)cn2cc(F)ccc2n1 60862,C(=O)(CCCS(N)(=O)=O)NC1CN(C(C(CCCOC)C)=O)CC1(C)C 60863,N1(C(C=C(C)c2ccccc2C)=O)CCC2C1CCCN2C(=O)C=Cc1cnc[nH]1 60864,C(=O)(CC1OCCc2ccccc21)N1C2CC(NC(C3CC3F)=O)CC1CCC2 60865,C1(CC(=O)NC(CC)CN(C)C(C2(CCOC)CC2)=O)SC(=N)NC1=O 60866,c1(C(=O)NC2C(NC(C(C)OCC)=O)C2)ccc2cccc([N+](=O)[O-])c2n1 60867,c1(OCC)ccc2ccccc2c1CN1CC2(CN(C(c3occc3C)=O)C2)C1 60868,CC(C(C)C(=O)N1CC(C#N)C1)NC(c1ccnn1CCF)=O 60869,c1(C(=O)NC2CN(C(CCCC(=O)NC(C)C)=O)C(C)C2)cnn2c1NCCC2 60870,N1(C(c2cc(C)[nH]n2)=O)CC2CS(=O)(=O)CC2(CNC(=O)CCC(C)(C)C#N)C1 60871,C1(NC(c2cccc(C(C)C)n2)=O)CCCCN(C(=O)C(=O)NCC2CC2)C1 60872,N1(C(CC2C(C)=NNC2=O)=O)CC(CNC(c2[nH]cnc2C#N)=O)C(C)(C)C1 60873,N1(C(CC2ON=C(CC)C2)=O)CCC(C(=O)NC(CC(=O)NC)C2CC2)C(C)C1 60874,c1(N(C2CCC(C)C2)C(C2(O)CN(C(=O)OC(C)(C)C)C2)=O)cnccc1.CO 60875,C(C(COC)C(=O)N1CCCC1CCC1CCCCN1C(c1ccsc1)=O)OC 60876,CC1CCCc2cc(C(=O)NCC3(NC(=O)CCN4CCCC4)CCOC3)nn21 60877,CC1(C2CCN(C(=O)CCC3CCCCN(C(=O)C4=NOCC4)C3)C2)CC1 60878,c1(NC2C(OC)C(C)(C)C2)nc2cccnc2c(=NCc2ccncn2)[nH]1 60879,S(=O)(=O)(c1cc(Cl)c(Cl)cc1Cl)NC(C1C(C(C)C)(CC)C1)=O 60880,c1(C(N2CCC(OCCNC(CC(CCC)O)=O)C2)=O)cnc(S(C)(=O)=O)s1 60881,c1(C(=O)NC(C2CCCCN2C(c2cnnc(O)c2)=O)C)nc(=O)n(C)[nH]1 60882,C12(CC)CCC(CC1)N(c1nc(C(F)(F)F)c(NC(C3CC3C(=O)OC)=O)s1)C2 60883,C1(C(N2CCN(C(CCCOC)=O)C(CCO)C2)=O)CCc2ccccc2O1 60884,C1(NC(CC2(C)CCN(C(C(C(C)C)OCC)=O)C2)=O)CC2CC1CC21CC1 60885,c1(C(=O)NC2CCN(C(c3c(SC)csc3)=O)CC2C)cnn2c1CC(F)(F)C2 60886,c1(C(N(CCC(=O)NC(C2CCOCC2)C#C)CCO)=O)ccc(C)cc1O 60887,C(N=c1[nH]c2cnc(Cl)cc2s1)C1(NC(C2CCC(=C)CC2)=O)COC1 60888,C(=O)(CC(C)C(C)C)NCC1(CNC(C2N(CC)CCC2)=O)CCC1 60889,N1(C(CC2N(C(C(C)OCCCC)=O)CC(O)C2)=O)CCC(F)(C#N)C1 60890,c1(C(=O)NC(C)(CNC(=O)C(=O)Cc2ccccc2)C2CC2)cccc(=O)o1 60891,C(CC(C)(C)CC(=O)NC(C1(O)CN(C(=O)CC(C)c2ccccc2)C1)C)OC 60892,C1(CN(C(=O)NCc2nnc(CC)o2)C)(SC)CCCCCCC1 60893,N1(C(CN(C(C(CCCC#C)C)=O)C2CCC2)=O)CCC2CCCC2CC1 60894,C1(CCC)CN(C(=O)CC2CCC(=O)N2C)CC1NC(C1(CC)CCC1)=O 60895,C=C(C)CC(C(=O)NCC1(C)CCCS1)NC(=O)CCOCCOC 60896,c1(C(N2C(C(N3CCCC(C)(O)C3)=O)C3CCC2C3)=O)n[nH]c2ccc(F)cc12 60897,CCC(C)(C(=O)NCC(CNC(C1(Cc2cccc(Cl)c2)CC1)=O)CO)OC 60898,N1(C(COC2CCN(C(c3n(COC)ncc3)=O)C2)=O)CCN(C)C(=O)C1CC 60899,CC1CN(C(=O)CCC2CCC(=O)N2)CC1NC(=O)C(c1ccc(F)cc1)F 60900,c1(CC)ccc([N+](=O)[O-])cc1C(=O)NCc1cccc(OCC2CCCO2)c1 60901,Cc1cc(C(=O)NC(C)C(C)(C)C(N2CC3CC(O)CC2C3)=O)ccc1C#N 60902,C(Cc1ccco1)(C(=O)N(C)Cc1cc(C)no1)NC(C=CC(CC)C)=O 60903,c1(C(N2CC(NC(C3(COC)CCC3)=O)CC2(C)C)=O)cc(Cl)c(OC)cc1Cl 60904,c1(CC)nc2n(n1)CC(NC(=NCCCF)NCC1(COC)CCN(C)CC1)CC2 60905,c1(CC)cc(C(=O)N(CC(C)NC(=O)C=Cc2nc(C)cs2)C)ccc1OC 60906,CC1CCN(C(=S)Sc2ccc(C(=O)NC(C)C(C)C(=O)O)o2)CC1 60907,CC(C)C(O)C(=O)NC(C1(O)CN(C(=O)CCNC(c2ncccc2O)=O)C1)C 60908,c1(CC)n[nH]c(=NC2CCN(C(c3cnn(-c4ccncc4)c3)=O)C(C)C2)s1 60909,N1(C(=O)OCC=C)CCN(c2ccnc(NCSC3CNC(=O)CO3)n2)CC1 60910,C=CCCCC(C(=O)OC)NCc1cc(Br)c(F)cc1OC 60911,c1(C(CNC(c2cnn(CC)n2)=O)NC(=O)CCC#N)ccccc1OC.C1CC1 60912,C1(C(=O)NC(C2CC(C(=O)NCCC(O)C3CCC3)C2)C)CCCN1C=O 60913,Cn1nnc2cc(C(N3CC4CCC4(NC(c4csc([N+](=O)[O-])c4)=O)C3)=O)sc12 60914,C1(C(=O)NC(CN(C(c2cnc(O)n2CC)=O)CC)C)CCCCC1(C)C 60915,C(C1c2ccsc2CCN1C(C1COC1)=O)NC(C(=O)NCC)=O 60916,Cc1cc(C(N2CCCCC2CS(N)(=O)=O)=O)ccc1Br 60917,S(=O)(=O)(c1cc(C)cnc1Cl)N1CCC(C(=O)Nc2cccc(C(C)=O)c2)C1 60918,C(=O)(C(=O)CCC(C)C)NC1(CC=C)CN(C(C2CC=CCO2)=O)C1 60919,C#Cc1ccnc(C(N2CCC(O)(CNC(=O)CC(COC)COC)C2)=O)c1 60920,Cc1cc(-n2nc(CO)nc2C(C)CN2CCC(N3CCCC3)CC2)ccc1Cl 60921,c1(OC)cccc(-c2cn(C3CCC(C(=O)NCC4CNC(=O)O4)C3)nn2)c1F 60922,c1(-c2onc(CN3CCC(O)(CO)C3)n2)cc2ccccc2c(O)n1 60923,C=CC1(C(=O)NCCCN2CC=CC2)CCN(C(=O)C(C2CCCCC2)C)CC1 60924,c1(C(=O)NC(CCCNC(c2c(NCC)scn2)=O)C)cnc2c(c1)CCCO2 60925,c1(SC)cnn(C)c1C(N1CC(NC(=O)CNS(N)(=O)=O)C(C)C1)=O 60926,c1(OC)c(C)csc1C(=O)N(C1CC(NC(=O)CCN(c2ccncc2)C)C1)C 60927,c1(-c2cc(OC)cc(F)c2C#N)cnc2[nH]cc(C(=O)N(C)C(C)C)c2c1 60928,c1(C(=O)NC(C)Cc2ccc(CNC(C3CC3C)=O)cc2)ccc(N)cc1F 60929,C1(CNC(C(n2cc(Cl)cn2)C)=O)CC2(CCC2)CN1C(C1CCCC12CC2)=O 60930,Cc1ccc(O)c(NC(c2nn(C)nc2Br)=O)c1 60931,CC1CN(C(=O)CNC(N)=O)CC1NC(c1cncc(C(C)(F)F)c1)=O 60932,CC(c1ccsc1)=CC(=O)NCCCC(C)NC(c1ccc(CO)s1)=O 60933,C(c1ccc(Br)cc1)=CCC(=O)NCCCCNC(C1CCC(F)C1)=O 60934,c1(C(=O)NC2(CCNC(=O)CCn3cc(Cl)cn3)CC2)cc(O)nc(O)n1 60935,Cc1cc(C(=O)NCCC(C)N(C)C(c2[nH]nnc2C)=O)cc(C)c1Cl 60936,C1(C(=O)NCC(C2CC2)NC(c2[nH]c(=N)sc2)=O)CC(=O)N(C2CC2)C1 60937,C1(CNC(C(CC=C)N(C)C)=O)COCCN(C(=O)C(=O)NC(C)C(=O)OC)C1 60938,C1(CN(C(C(C)n2ccnn2)=O)C)CCCN1C(C1CCCN1C1CC1)=O 60939,C1(C(=O)NC(C2CCOC2)CC)(CNC(c2ccns2)=O)CCCC1 60940,c12ccc3c(n1)CN(C3)C(=O)N2.C1(CCNC(c2ccccc2)=O)CCOC1=O 60941,c1(NCC)cnccc1C(=O)N(CCNC(C1CC1(C)C(C)C)=O)C1CC1 60942,C#Cc1ccc(CC(=O)NCC=CC(=O)NCC(C)C)cc1 60943,c1(C(N2CCC(O)(CNC(C(C(C)C)SC)=O)CC2)=O)ncnc2c(C)csc12 60944,Cc1ccc(C(C)(C)C(N2CCCC(C(=O)NC3CN(S(C)(=O)=O)C3)C2)=O)cc1 60945,c1(C(=O)NCC2N(C(COC)=O)CC=C2)cccc(-n2cccn2)n1 60946,C1(C(=O)NC(CC=C)CO)CC2(CCN1C(C1CCCC(C#N)C1)=O)CC2 60947,C(c1cccc(Cl)c1)=CC(=O)N(C1CCN(C(c2c(C)coc2)=O)C1)CCO 60948,C1(CC(=O)NCC(CO)NC(C(C)C2CCC2)=O)CCN(CCF)CC1 60949,C1(C(N(CC(CNC(CN(C(C(C)C)=O)C)=O)C)C)=O)CN2CCN1C(C)C2 60950,C(N=c1cccc(S(=O)(=O)NCC=CBr)[nH]1)C1C(c2ccc(C)cc2)CCC1 60951,N1(C(C2(CCC)CC2)=O)CCC2(CO)CN(C(=O)CC3(O)CCCCC3)CC2C1 60952,Cc1nc(Cl)[nH]c(=NCC2C3CN(C(=O)C(C)Cc4ccc(F)cc4)CC23)c1F 60953,C(=O)(C(O)CNC(=O)CN1CC=CC1)NC(C#C)CC1CCCC1 60954,C12(CNC(C(CC=C)(F)F)=O)CCC(CNC(C3(C)CC3(F)Cl)=O)(CC1)CO2 60955,c1(C(=O)NC23CC(NC(c4nccc(C=C)c4)=O)(C2)C3)cccn2ccnc12 60956,CC(CC(F)F)C(=O)N1CCCC(O)(CN(C(=O)CC2CCSCC2)C)C1 60957,N1(C(C2CCCO2)=O)CC(n2cc(C3CCCO3)nn2)C(O)C1 60958,C1(CNC(=NCCOC)NCC2=CCOCC2)CN2CCCCC2CO1 60959,C12(CNC(NCC3(COC)CCCCO3)=NCC(C)C)CC3CC(CC(C3)O1)C2 60960,N1(C(Cn2c(C)ccn2)=O)CC(C)CN(C(=O)C2=CSCCO2)C(C)C1 60961,[N-]=[N+]=NC1CC2(C(N3CC(O)(CCNC(C4(Cl)CC45CCC5)=O)C3)=O)CC12 60962,N1(C(C(C)OCC2CCCO2)=O)CCC(NC(C23CCC2C3)=O)CC1 60963,C(=O)(C(C)(C)CC(C)C)NC1(CNC(C(C)SC)=O)CC1 60964,C=Cc1ccc(CN2CC3(CN(C(c4ccccn4)=O)C3)C2)cc1 60965,C(=O)(C1CCCn2nccc21)NCC1CCC2(CN(C(C3CC(=O)NC3)=O)C2)O1 60966,O=CN1CCCC1C(N1CC(O)CC1CNC(=O)C(O)c1ccco1)=O 60967,Cc1nc(CC(N2CCC(C(C)(C)NC(=O)CCC3CSCCS3)C2)=O)cs1 60968,c1(OCCCC)ccc(S(=O)(=O)NC2CC(S(C)(=O)=O)C2)cc1N(C)C 60969,Cc1cnc(C)c(NC(C2CC(F)CN(C(c3ccc(Cl)c(Br)c3)=O)C2)=O)n1 60970,C1(NC(c2cnc(C)o2)=O)CCN(C(C2CC23CCSCC3)=O)C1(C)C 60971,S(=O)(=O)(c1ccc(Br)cc1NCCc1ncccn1)N(CC)CCO 60972,N1(C(C2C(C)C2C)=O)CC(NC(c2cc(N)nc(Cl)c2)=O)CC(C)(C)C1 60973,c1(OC)ccc(CN2CC(CNC(c3ncoc3C)=O)C2)nc1Br 60974,C1(C(=O)NC(C)CCN(C(=O)CCc2ccco2)C)CC2(C1)CC2F 60975,C=CC(C)(O)C(=O)NC(C1CN(C(c2ccnc(SC)c2)=O)CCO1)C 60976,N1(C(CN(c2ccccn2)C(C)=O)=O)CC2CC1C2CNC(c1c(C)ccn1C)=O 60977,CN1CC2CCN(C(=O)CC3CCCCN3C(=O)CNC(N)=O)CC2C1 60978,CN1CCCC(CCC(N2CC(NC(c3ocnc3C3CCC3)=O)C(O)C2)=O)C1 60979,c1(C(=O)NCC(CN(C)C(C2(C(F)(F)F)CC(C)(C)C2)=O)O)cn2c(n1)CCC2 60980,c1(C(=O)NC(CC=C)CNC(=O)C(O)CC(N)=O)cc2sc(Cl)cc2[nH]1 60981,C1(NC(C2(CC)CCC2)=O)CCN(C(=O)CSCCN(C)C)CCC1CO 60982,N1(C(COCCCC)=O)CC(C(N2CCCC(C(C)(C)C)C2)=O)CC1(C)C 60983,CCCCS(=O)(=O)NC(C)C(=O)NCCCN(C(=O)CC1(CO)CC1)C(C)C 60984,c1(CNC(=O)NCc2c(CS(=O)(=O)NC)cccc2)cnc(Cl)cc1Cl 60985,c1(CC(=O)NCC(C)N(C(c2ccnnc2)=O)CC)cc(Br)cnc1OC 60986,C=Cc1cncc(C(N2CCC(N(C(=O)CNS(=O)(=O)NC)C(C)CC)C2C)=O)c1 60987,C1(CNC(C(C)OC(C)=O)=O)CC(C(=O)NCCN2CC=CCC2)CO1 60988,c1(OCC(N2CCC(C)N(Cc3ccccc3)CC2)=O)ncnc2ccccc12 60989,CCC(C(=O)NC1CC(CN(C(=O)C(C)N(C)C)C)C1)C(C)(C)CC 60990,C(CC(C(=O)NCCC=CCCC)NC(c1cc(C2CC2)on1)=O)=CC 60991,O=C(C1=CCCOCC1)NC(CNC(C1(F)CC1c1ccccc1)=O)CO 60992,CC1CCC(CNC(=O)Cc2cncnc2O)CN1C(c1cc(=O)n(C)cn1)=O 60993,CCC(C)C(O)C(C)C(=O)N1CC2CCC1CN2C(=O)CN1C(=O)CNC1=O 60994,Cc1c(C(N2CC(NC(=O)C(C)OCCN(C)C)C2)=O)nn2c1OCCC2 60995,N1(C(C(C)CC2CCCC2)=O)CC2CC1CC2NC(C1(C)COC1)=O 60996,C(=O)(C(=O)N=S(C)(C)=O)NCCC1CN(C(=O)C=Cc2ccsc2)CC(C)O1 60997,c1(C(N2C(C(N3C4CCCC3COC4)=O)CCC2)=O)cc(Br)cc(Cl)c1F 60998,C1(NC(c2n[nH]c(C3CC3)c2Br)=O)CCCCN(C(=O)CC2CCCC2)C1 60999,c12ccc(Br)c(c1C)NC(=O)N2.C1(C(=O)OC)(C(=O)OC)CCCO1 61000,N1(C(=O)CCCF)CCCC2C1CCCN2C(=O)CSCC(F)(F)F 61001,C1(NC(=O)Cc2ccccc2C2CC2)CCS(=O)(=O)C12CN(C(=O)CC1CC1)C2 61002,CCC(CC(=O)NCC(C)NC(c1ccnc(C2CC2)n1)=O)C(F)F 61003,N1(C(CC2(CC=C)CCCC2)=O)CCCC1(C)CNC(C12CCCC1C2)=O 61004,c1(CCC(=O)NC(CC2CN(C(C(COC)OC)=O)C2)C)cccc(F)c1 61005,CCCCCC(O)C(=O)N1CC(C(O)C(=O)Nc2ccc(N(C)C)nc2)C1 61006,N1(C(C=C(CCC)C)=O)CC2CC(NC(=O)C=Cc3cccs3)CC(C2)C1 61007,C(C(=O)NNC(=O)C(F)(F)F)C(c1c(C)cc(C)c(C(C)=O)c1C)=O 61008,Cc1nc(C)n(CC(=O)NC2COCCC2C(=O)N(C)CCC2CCCN2C)n1 61009,N#Cc1ccc(C(F)(F)C(N2CCOCC2Cc2nn[nH]n2)=O)cc1 61010,C(=O)(C(C)(C)C(=O)NCC(C)NC(c1ccc(SC(F)(F)F)s1)=O)OCC 61011,c1(C(N2CC(CC)(NC(=O)CC3CC(=O)NC3=O)C2)=O)cncc(F)c1C 61012,N1(C(c2sccc2Br)=O)CC2(C1)CN(C(c1ccc(O)cc1F)=O)C2 61013,Cc1cc(CCC(=O)NCC(C)(C)CN(C)C(C2CCN(C)C2)=O)nn1C 61014,C(=O)(C(F)CC(C)(C)NC(c1ccccc1)=O)N1C(C)(CC)CC1 61015,C(CC(C)(C)NC(c1cnco1)=O)N(C(=O)CCSC1CCCC1)C 61016,C1(NC(c2n(C)ncc2)=O)CCN(C(c2cccc(C(F)(F)F)c2O)=O)CC1F 61017,C1(NC(=O)COCCCF)CN(C(c2cnc3ncccn23)=O)C2(CCCC2)C1 61018,C(=O)(C(C)(C)C)NC(C)C(=O)N(C)CCNC(C1(CC2CC2)CCCO1)=O 61019,Cn1c(O)ncc(C(=O)NCC2CCC(NC(c3cc(C(F)F)[nH]n3)=O)C2)c1=O 61020,c1(NC(N2CCN(Cc3ccccc3)C(c3cccs3)C2)=O)ccc(Br)cc1Br 61021,n1(C(C(C)O)C)cc(C2(O)CN(C(=O)C(c3ccccc3)F)C2)nn1 61022,C1(NC(CS(=O)(=O)NC)=O)CCN(C(=O)C(n2cc(Cl)cn2)C)CC1O 61023,c1(CC(=O)NCC(CNC(Cn2c(C)c(Cl)cn2)=O)C)cc(C(F)(F)F)cc(F)c1 61024,C1(NC(COCc2ncc(C)o2)=O)CCC(C)(CNC(=O)CCc2ccsc2)C1 61025,c1(C(=O)NC2C(CNC(c3cn(C(C)C)nc3)=O)CC2)cccc2c1CCCC2 61026,N1(CCO)CCN(CC(c2ccccc2)F)CC1.c1(C(CO)N)ccccc1 61027,C(=O)(C(C)(CC)OC)N1CC(CC(C(=O)NC(CC)(C2CC2)C2CC2)F)C1 61028,C1(C2CCN(C(=O)Cc3cc(Cl)ccc3Cl)CC2)(NC(C2CNC(=O)N2)=O)CC1 61029,C1(C(=O)NCC2CCCCN2C(=O)COCCCF)CC2CC1CC2(F)F 61030,c1(OC(C)C)ccccc1CC(N1CC(N(C)C(c2cscn2)=O)C(F)C1)=O 61031,O=C(CC1COc2ccccc21)NC1CC(NC(=O)C(F)(F)c2cncs2)C1 61032,C(=O)(CC(C(F)F)C(C)(C)C)N1CCC(CCNC(C2=C(C)CCC2)=O)CC1 61033,c1(C(N2CCC(N(C(C(C)OCC=C)=O)CCO)CC2)=O)ccc(F)cc1C 61034,N1(S(CCC)(=O)=O)CCC(C(N2CCC2CNC(=O)CCC(C)OCC)=O)CC1 61035,C(=O)(C(O)C(F)(F)F)NCCC1CC(NC(C(C)Sc2ccccc2)=O)C1 61036,CCC(CC(=O)N(CC(=O)N(C1(c2cc[nH]n2)CC1)C)C1CC1)SC 61037,C1(N(C(=O)CN(C)C2CC2)CC#C)CCN(C(C2(C(=O)OC)CC2C)=O)CC1 61038,N1(C(CNC(=O)NC)=O)CCC(CO)C(NC(=O)CN2CCC(C)(C)C2)C1 61039,Cc1cc(=NCc2cnccc2C)[nH]c(=NCc2ccn3ncnc3c2)[nH]1 61040,c1(OC)cc(C(=O)NC2CC(NC(=O)CC(C)(C)SC)C(O)C2)cc(C)c1 61041,c1(CC)c(C(=O)NC(C)CCCNC(c2conc2C2CCC2)=O)cccc1C 61042,C1(CNC(=O)COC(CNC(CN(C)C2CC2)=O)=O)CC(NC(C)(C)C)C1(C)C 61043,C(CC(C)C)(C(=O)N1CCC(CNC(c2nnn(C(C)(C)C)n2)=O)C1(C)C)OC 61044,CC(C)CCC(C)N=c1[nH]c(=NCC2CCC=CO2)[nH]c2c(F)cccc12 61045,CC1(C(=O)NCC(C2CCOC2)NC(c2cnc(N(C)C)cn2)=O)CCCCC1 61046,c1(-c2n(CC=CC)c(N3CCCOC3C)nn2)csc(=Nc2ccccc2)[nH]1 61047,C1(CC)CN(C(=O)Cn2ncnn2)CCN1C(=O)Cc1cc(O)ccc1Br 61048,C1(CNC(C=C(C)C)=O)(CNC(=O)Cn2cnc([N+](=O)[O-])n2)CC2CCCC2C1 61049,c1(OCC(CC)CNC(=O)C(n2cc(CCC(C)(C)O)nn2)C)cccc(C)c1 61050,C1(C(=O)NC(C(CO)NC(CCSCC(=O)OC)=O)C)CC(C)c2nc(C)cn2C1 61051,c1(OC)csc(C(=O)N(C2CCC(NC(C3(n4cccn4)CCC3)=O)C2)C)c1 61052,C12(NC(=O)NCCC(C)(O)C3CC3)CC1CS(=O)(=O)C2 61053,N#Cc1sc(=NCC2CCN(C(c3cc(Cl)no3)=O)C2)[nH]c1Cl 61054,C1(NC(C2OCCN(C)C2)=O)CC2(CCN(C(c3ccc(C#N)c(O)c3)=O)C2)C1 61055,c1(NC(C2CC2)=O)cc(CC2CC2)ncn1.O=C1CSC2(CC2)CCN1 61056,C(=O)(C(CCC)CCCO)N(CCCCC)CC1CCC2CC2CC1 61057,c1(C(N(C)CCNC(C2CCCN(C(=O)CNC=O)C2)=O)=O)ccccc1[N+](=O)[O-] 61058,CCCCC(CC)CC(=O)N(CC(C)NC(c1ccn(CC)c1C)=O)C 61059,c1(C(N2CCC(CNC(C(C(C)C)F)=O)C2(C)C)=O)nccc2cccnc12 61060,Cc1noc(-c2cn(CC(=O)NCC(C3CC3)N(C)C(c3ccon3)=O)cn2)n1 61061,C1(CNC(CCCSC)=O)CSCCN1c1nccc(CC#N)n1 61062,CS(C)(=O)=Nc1ccc(C(N2CC3CCCC3(CNC(C3(F)CC3)=O)C2)=O)cc1 61063,Cn1cnc(NC(=O)NCC2(c3cccc(C(F)(F)F)c3)CCC2)cc1=O 61064,N1(C(c2ccc(C)o2)C(=O)NC2(CC3CC3)CCC2)CCn2c(C)nnc2C1C 61065,C=CCC(C(=O)OCC)NC(=O)CCN(C(C1CCC1C)=O)CC1CC1 61066,C(=O)(CCC(C)C#N)NCC1N(C(c2c(C)coc2C(C)C)=O)CCC1 61067,c1(C(=O)NCC2(OC)CCN(C(=O)C=Cc3cccnc3)C2)cc(C)c(C)cn1 61068,C(=O)(CCCCC(C)C)NC(CCC(=O)NCCc1nc(C)sc1)C 61069,Cc1[nH]nc2c(C(N3CCC(CO)(NC(C4CNC(=O)N4)=O)CC3)=O)cccc12 61070,N1(C(C2CN(C(CNC(N(C)C)=O)=O)CC(F)(F)C2)=O)CCC2(CCOC2)CC1 61071,C(N=c1[nH]c(=NCC(C)(F)c2ccccc2)c2[nH]ccc2[nH]1)C1C(C)(C)C1 61072,C(C1CCC(C)CC1)=C(C)C(=O)NC1CC(C)N(C(C2CC(=O)CO2)=O)C1 61073,c1(OCC)ccc(CC(N2CCC(NC(=O)C=CSc3ccccc3)C2)=O)cc1 61074,N1(C(CC(CC)C)=O)CC2CCCN(C(=O)C=Cc3nc(C)co3)C2C1 61075,C1(C(N2C(C(=O)NCc3ccn(C)n3)COCC2)=O)CCCCCCC1 61076,C1(NC(C2CN(CC)C(=O)C2)=O)CCC12CN(C(c1cn(CC(N)=O)nn1)=O)C2 61077,CC1(C)C(CN(C(=O)Cn2ncnn2)C2CC2)CCN1C(C1CC1c1ccco1)=O 61078,C12(NC(CCc3cnc(C)o3)=O)CCN(C(c3ccn(C)c3)=O)CC1C2 61079,c1(OC)cc(Nc2ncc(Cc3ccc(C(C)(C)C)cc3)s2)ncn1 61080,c1(C(=O)NCC(C)NC(=O)C(F)CC2CC2)ccc(Br)cc1 61081,c1(CC)nn(C)c(Cl)c1C(=O)NC1C2CN(C(c3coc(OC)n3)=O)CC12 61082,Cc1nn(CCO)c(C)c1C(N1CCC(c2ccnnc2)CC1)=O 61083,CC1CN(C(c2cc(O)cc(O)n2)=O)CCN1C(c1ccsc1Br)=O 61084,c1(C(=O)NCC(C(=O)Nc2c(CC)ccnc2)(C)CC)ccc2nccn2c1 61085,C1(NC(=O)NCC2(CC)CCCO2)CC2CC1CC2C(=O)O 61086,C1(NC(C2N(C)C(=O)CC2)=O)CN(Cc2ccnc(F)c2Cl)CC1C#N 61087,N1(CCN(CC)CC)CCCCC1C1(NC(=O)COCC(C)C)CC1 61088,N1(CCC#C)CCN(C(=O)NC2C3CCC(F)C23)CC1 61089,C(=O)(CS(=O)(=O)Cc1cncn1C)NC(c1ccc(Cl)cc1)C(C)C 61090,CC1CC(C)N(C(c2cccc3oncc23)=O)CCN1C(c1ccco1)=O 61091,N1(C(C2C(C=C)OCC2)=O)CCN(C(c2c(C(C)C)nn(C)c2Cl)=O)CC1CC 61092,C1(NC(C2CCC(C)O2)=O)CCC2CN(C(=O)C(c3ccccc3)C)CCC2C1 61093,c1(CC(N2CC(C(N)=O)(CNC(C3C(C)C3C)=O)C2)=O)cccc(Br)c1 61094,N1(C2CCC(NC(COCCCCC)=O)C2)CCN(C(=O)C(Cl)=CCl)CC1 61095,CC(C)=C=CC(=O)N(CC(O)CNC(=O)COC1CC1)C 61096,C1(CNC(C(CC#C)C2CC2)=O)CC2(CCC2)CN1C(c1ccnc(CO)c1)=O 61097,N1(C(CCOCCC)=O)CC(NC(C2CC(Cl)(Cl)C2)=O)CC12CCC2 61098,C(=O)(C(C)S(C)(=O)=O)NC1C(CC)N(C(=O)CCn2ccnc2)CC1 61099,N(C1CCCc2cc(C#N)ccc21)Cc1cc(CC(OC)OCC)no1 61100,C(C(C)C(F)C(=O)NC(C)C(C)SC)NC(C1(C(=O)OC)CC1)=O.C(C)(=O)O 61101,C(=O)(C1=CC2CCCC12)N1CCCC(C)(NC(C(c2c(C)noc2C)C)=O)C1 61102,Cc1onc(C(F)(F)F)c1C(=O)NC1CCN(C(=O)CN2C(C)CCC2C)CC1 61103,Cc1ccc(=O)n(CC(=O)NCCCCNC(=O)C(c2ccc(F)cc2)(C)F)n1 61104,CCC(C)(C)C(C)CNc1ccc(OCc2cccs2)cc1 61105,C1(C(=O)OC)C(NC(=O)NCc2cccnc2C)CCN1C(=O)Cc1ccon1 61106,CC(CCN=c1[nH]c(=NCc2csc(N(C)C)n2)c2[nH]ccc2[nH]1)CC(C)(C)C 61107,CCCC(C)(O)C(=O)NC1CCC(CNC(=O)CCn2cnccc2=O)CC1 61108,C1(Cl)(C(=O)NCCNC(c2cnc(C(F)F)s2)=O)CC12CCOCC2 61109,C12(CNC(C3(CC)CC3)=O)CCCCC1CN(C(c1ccc(CSC)cc1)=O)C2 61110,Cc1nc(C=CC(=O)NC2CC23CC(NC(=O)CCNC(N)=O)C3)[nH]c1C 61111,c1(C(=O)NCC(C)CN(C)C(c2cnn(CC(F)F)c2)=O)cc(C(N)=O)c[nH]1 61112,c1(C(N2C(C)CN(C(c3cc(SC)oc3)=O)C(C)C2)=O)ccc2c(c1)N(C)CC2 61113,C1(C(=O)N(CC(O)CN(C(=O)Cc2n[nH]cc2Br)C)C)(OC)CCCCC1 61114,C(=O)(N=c1[nH][nH]c2c1CN(C(c1c(F)cc(Br)c(F)c1F)=O)C2)C1C(C)(C)C1 61115,CCC(C)C(C(=O)NC1CC(F)(F)C1)N1CCC(C(=O)NCCC#N)CC1 61116,C1(C(=O)NCC2CCN(C(c3ccccc3O)=O)C2)CCC2C(CC1)C2(F)F 61117,C1(NC(Cc2c(C)ccs2)=O)CCCC(NC(=O)CC(=O)N(C)C)CC1 61118,C12(C(=O)NCC(C(CC)C)C)CC(CO1)N(C(C1CCC(C)(C)OC1)=O)C2 61119,c1(C(N(CCOC)CCNC(=O)C(O)C2CCC2)=O)cc(P(C)(C)=O)cs1 61120,c1(C(=O)NCC(C)N(C(c2c(NCC)scn2)=O)C)c[nH]c2ccc(F)cc12 61121,c1(C(N2CC(CNC(CC(CCC)O)=O)CC2(C)C)=O)ccc(N)cc1[N+](=O)[O-] 61122,C1(NC(C(C(C)C)O)=O)CCC(C)(CNC(c2nn(C)cc2Br)=O)CC1 61123,CC(C)C(C)C(=O)NCc1cc(C(=O)NOCC2CCOC2)on1 61124,Cc1ccc(C(=O)NCC(c2ccccc2)CNC(=O)CC#N)c(F)c1 61125,n1(CCC)cc(Cl)c(C(=O)NC2CCC(C)(CNC(C3CN(C(C)=O)C3)=O)C2)n1 61126,C1(CC(C(=O)NCCCF)N(C)CCn2cncn2)CCC(C)(C)O1 61127,Cc1ccccc1C=CC(=O)NCC1(C(=O)N(C2CCCC2C)C)CCC1 61128,c1(C(=O)NC2CC(NC(C3CCC(C)S3)=O)C2)cc2sc(Cl)cc2s1 61129,N1(C(C(CC)NC(N)=O)=O)CC(NC(=O)C#CC(C)C)C(C)C1 61130,C(c1cc[nH]n1)=CC(=O)NCC(C)(C)OCCNC(C1CCCC1O)=O 61131,Cc1cccc2c1OCCC2NC(=NCCN1CCCC1C)NC1CC1 61132,CC(O)(C(=O)N1CC(C(=O)NCCN2CCC(O)C2)C2(CCC2)C1)C(F)(F)F 61133,C#CCC(C(=O)NCC(N1CCOCC1)=O)NC(=O)C(F)OC(F)(F)F 61134,C1(CC)CCN(C(c2cscc2Cl)=O)C1C(=O)NC1(CC(N)=O)CC1 61135,c1(CN2CC3C(NC(=O)Nc4c(C)ccc(C)c4)C3C2)ccc2c(c1)CCC2 61136,CC1(C)OC2(Cn3nnnc3N3CCN(c4cncc5nccn45)CC3)CCC1C2 61137,C(=O)(C(CCC)C(C)C)N1CC(NC(CCC=CC)=O)C2(C1)CC2 61138,N1(C(C(C(C)(C)C)OC)=O)CC2(CC(NC(=O)CSCc3ccccc3)CO2)C1 61139,C(C)(CNC(c1cn(-c2ccn(C)n2)cn1)=O)(CO)NC(C=C(C)C)=O 61140,c1(CCCC(=O)N(CCCCNC(c2occ(C)c2)=O)C)c[nH]c2ccccc12 61141,CCCC(C)(CC)C(=O)N1CCC(CN(C(=O)CSCC(=O)NC)C)C1 61142,CC1(C)CN(C(c2sc(C#N)cc2Cl)=O)CC(CNC(c2n[nH]cc2F)=O)O1 61143,Cc1c(C(=O)NCC2(NC(=O)C(C(C)C)NC(N)=O)CCOCC2)cnn1C 61144,C(CC(=O)N1CCC(CC(N)=O)C1)(C(C)(C)C)NC(Cc1ccc(C#C)cc1)=O 61145,N1(C(COc2c(C)ncnc2C)=O)CCN(C(C2CCC(O)C2)=O)CC(C)(F)C1 61146,Cc1cc2c(C(=O)N(C(C)CCNC(C3CCNC(=O)C3)=O)C)cccc2o1 61147,c1(C(=O)NCC2C(CNC(=O)CCc3cocn3)C2)cc2occc2s1 61148,c1(C(=O)NC2CCN(C(C(C)(C)NC(=O)OC)=O)C2)cc(C)nc2cc(C)nn12 61149,C1(CNC(C2C(CNC(C(CC#C)O)=O)C2)=O)CCC2(CC2)CO1 61150,c1(C(=O)NC2C(NC(C(C(=O)OC)C)=O)CC2)cnc2cc[nH]c2c1 61151,C(=O)(C1=NOC(C)C1)NCCCN(C(=O)CN(CC)Cc1ccccc1Cl)CC 61152,c1(C(N(C)CC2CCCN(C(CC(COC)C)=O)C2)=O)c(OC)cccc1F 61153,C#Cc1ccc(OC)c(C(N2CC(CNC(=O)C=CSC)CC23CCC3)=O)c1 61154,Cc1cc(C(=O)NCCCN(C(c2ccc(C(F)F)s2)=O)C2CC2)[nH]c1C 61155,C1(C(N2CC3C(NC(C(CCC)Cl)=O)C3C2)=O)CC2(CCC2)CO1 61156,C1(NC(c2ccc(N(C)C)cc2)=O)CC2CC1CN(C(c1cc(Cl)no1)=O)C2 61157,c1(C(=O)NC(C(C)C)(C)CNC(=O)C(C)CC(N)=O)ncsc1S(N)(=O)=O 61158,CCS(=O)CC(=O)NCC1CCCC(CNC(C2(n3cccc3)CC2)=O)C1 61159,C(=O)(C1CCc2cccnc21)NCC(CCNC(c1ncn(C)n1)=O)O 61160,C=C(Cl)CCC(=O)N1CCCC(CN(C(=O)CC2OCCC2C)CC)C1 61161,N1(C(c2cc(C)n(C)c2)=O)CC2(CCN(C(c3ccc4occc4n3)=O)CC2)C1 61162,C#CCCCC(=O)N1CCN(c2ccccc2NC(C2CC=C(C)CC2)=O)CC1 61163,Cc1ccc([N+](=O)[O-])cc1-c1nc(C(=O)Nc2c(O)cccc2C#N)ccc1F 61164,c1(CN2C(C(N3CC(F)C(F)C3)=O)CC3CC32)c(F)cc(F)cc1Br 61165,C(C)(CCC(=O)NC(CCC1CCC1)C(=O)NCCc1ncccc1F)OCC 61166,CC1(C)CC(NC(=O)CC2CC3(C2)CN(C(=O)CC2(C)CC2)C3)C(=O)O1 61167,c1(CC)ccc(C(N2CCCN(C(C3(F)C4CCCC34)=O)CC2)=O)cc1CC 61168,c1(CS(C)(=O)=O)oc2ccccc2c1NC(c1csc2ccc(Cl)cc12)=O 61169,N1(C(CN2CCC(C)C2)=O)CCC2(CC2)CC1C(=O)Nc1cnc(Cl)nc1 61170,c1(C(=O)NC(CNC(C(CCCC#C)C)=O)C)cnc2[nH]c(C)nc2c1 61171,c1(-c2ccc3[nH]nc(C(=O)NCCNC(C)=O)c3c2)nc2cc(C)cc(C)c2[nH]1 61172,CCC(CC)C(C(=O)N1CC2(C)CC1(C(N1CCCCC1CC(C)C)=O)C2)OC 61173,C=CC(C)(CC)C(=O)NCC1=CCN(C(=O)C(C)c2cncs2)CC1 61174,CCCCC(C(=O)NCC1(O)CCCN(C(c2cnn(CC)c2)=O)C1)N(C)C 61175,C1(NC(C(CCC)NC(N)=O)=O)CC2CC1CN(C(=O)CCCCC(C)C)C2 61176,CC1(C)C(c2cn(Cc3cccnc3)nn2)CCN1C(C1CCN1C(C)(C)C)=O 61177,C=CCC(C(=O)NC(CO)CCCCNC(=O)CN(C)C(=O)OC)C(C)C 61178,CC(C)(CC1CCOCC1)C(=O)NCC(C1CCCC1)NC(C1CC(CF)C1)=O 61179,c1(CCOCC(N2CC(CC(C)NC(c3cnc(S)[nH]3)=O)C2)=O)ccccc1 61180,C1(C(N2C(C)CC(NC(c3cc(CC)n(C)n3)=O)C2)=O)CN2CCC1CC2 61181,CC1CN(C(=O)CC2(C)CCCCC2)CCC1CNC(C1(C)COC(=O)N1)=O 61182,C(=O)(C#CC(C)(C)CNC(=O)CC1(COC)CC1)NC(CCCC=C)C1CC1 61183,C1(O)(C(C)NC(CCC(=O)c2ccc(C)s2)=O)CCN(C(C2CCCS2)=O)CC1 61184,N1(CCNC(C2CCCC23CC3)=O)CCN(C(=O)CN2CCCS2(=O)=O)CC1 61185,c1(C(N(C2CCCN(C(=O)CCc3ncc[nH]3)C2)C)=O)cnc2c(Cl)cccn12 61186,S(=O)(=O)(CCC(=O)NC1CCN(C(=O)Cn2cnc(Br)c2)C1)N(C)C 61187,c1(C(=O)NCC2N(C(COCC)=O)CCC2C)ccc2c(c1)N(C)CCO2 61188,N1(C(Cc2c(C)ncs2)=O)CCCC2(CCN(C(C3CN(C4CC4)C3)=O)CC2)C1 61189,c1(C(N2CCC(NC(C3(C)CCCNC3=O)=O)C2)=O)cccc2c1OCCCO2 61190,N1(C(=O)CSc2nc[nH]n2)CCCC2(C1)CN(C(c1cnc(O)s1)=O)CCO2 61191,Cc1nc2c(C(=O)NC(C3(CNC(c4sncc4C)=O)CC3)C)cccc2o1 61192,N1(C(c2c(CC)n(-c3ccccc3)nn2)=O)CCC2(CC1)CC(O)(C(F)(F)F)C2 61193,CCC(CC(=O)O)N(C(=O)C(C)CN(C)C)C.C1(C(=O)O)CC(C(F)F)C1 61194,Cc1oc(C)c(C(=O)NCC23CC(CN2C(=O)Cn2cc(F)ccc2=O)C3)c1C 61195,Cc1cc(OCc2ccc(C(=O)NCC(C3(C)CCC3)O)cc2)ccc1[N+](=O)[O-] 61196,C(C)(CCC(=O)NC(C)(CNC(=O)CSCC(N1CCCCC1)=O)CO)OCC 61197,CCCCC(C)(F)C(=O)NC1CCN(C(c2ccc(COC)o2)=O)CC1CC 61198,C1(C(=O)NC23CN(C(CCOCC(C)C)=O)C(CC2)C3)Cc2c(F)cccc2O1 61199,c1(C(=O)NCCCCCN(C(C2CN(CC(C)C)C2)=O)C)cc(F)ccc1O 61200,C(=O)(C1COc2ccccc21)NC(c1ccc(N(C)C)cc1)CNC(=O)CO 61201,C(=O)(C1=CCCCC1C)NC1(CNC(C2CCN(CC(C)C)C2)=O)CC(F)(F)C1 61202,C1(COC)CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CCN1C(C12CCC(F)(CC1)C2)=O 61203,CC(C)CC(CNC=O)CC(=O)NCC(C)N(C)C(c1cccc2nonc12)=O 61204,N1(C(c2c(OC)c(Cl)sc2)=O)CCCC2(NC(C3CN4CCC3CC4)=O)CC2C1 61205,Cc1nc(C2CC2)[nH]c1C(=O)NC1CCCC1NC(=O)CC1CCC(C)(C)C1 61206,C1(CNC(c2c(CC)cno2)=O)CC2(CC2)CN1C(c1ccc(Cl)c(OC)c1)=O 61207,C12(CCCCC1)CC(=O)N2.C(c1cocn1)=CC.C1CCCCCOCCN1CC 61208,C12(C(=O)NCCc3nccc(C)n3)CC(CN(C(=O)CCCC#N)C1)C2 61209,C1(NC(CCCOCC=C)=O)CCCCN(C(=O)Cn2cc(C)ccc2=O)CC1 61210,CCCCC(C(=O)NCC1(CC2CC2)CCC1)NC(=O)C1=CC(C)(C)C1 61211,c1(OC)ccc(C(N2CC(NC(C3CC(CN(C)C)C3)=O)CC2C)=O)nc1Cl 61212,Cc1ncc(Cl)cc1C(=O)NCCOCCNC(=O)C(F)(F)c1cnn(C)c1 61213,N1(C(c2ncc(C)o2)C)CCCC(C(N)=O)(NC(=O)CN2CCCCCC2=O)C1 61214,N1(C(c2c(OCC)nccc2)=O)CC(NC(=O)CCN(C)C(C)=O)CC(F)(F)C1 61215,Cc1ccnnc1C(N1CCC(Cn2cc(-c3ccc(Cl)s3)nn2)C1)=O 61216,C(CC(=O)NCC(C)S(N)(=O)=O)(CC(C)C)NC(C1N(C(C)=O)CCC1)=O 61217,C(=O)(CC(C(F)(F)F)NC(C1CCCN1C(N)=O)=O)NC1CC(C)OCC1 61218,CCC(C)CCC(=O)NCC1(OCC)CN(C(c2cc(=O)cc[nH]2)=O)C1 61219,N1(C(C(C(=O)OCC)(C)F)=O)CC2(CCC(NC(=O)Cn3ccnc3C)CC2)C1 61220,c1(C(=O)NCC2CCN(C(Cc3cn(C)nn3)=O)C2)cc(C(F)(F)F)ccc1Cl 61221,c1(C(=O)NCC2CC(N)C2)ccc(S)nc1.CC(C(=O)SC(F)(F)F)OC(C)(C)C 61222,C12(NC(c3nn(C)c(CO)c3)=O)CCCC(NC(=O)C=CCOC(C)(C)C)(C1)C2 61223,C1(NC(C(C)=CC2CC2)=O)C2COCC1CN(C(c1nnc(O)nc1O)=O)C2 61224,N1(C(c2c(C)nc(Cl)cc2)=O)CCOC2(CCN(C(c3ccon3)=O)C2)C1 61225,CC(C)C(CNC(=O)Cc1ccc(F)nc1)C(=O)NC1CCCC(O)C1 61226,CCCCC(=O)C(=O)N(CC(N1CC2C(N(C)C)C2C1)=O)C 61227,CC1=C(C(=O)N2CCCCC(CNC(C3CCC3)=O)C2)CCC1 61228,C(=O)(C(N)CCCCC#N)N1CCCC(N(C)C)CC1 61229,C1(C(=O)NC2(CO)CN(C(c3c(OC)cc(C)s3)=O)C2)CCc2nnnn2C1 61230,n1(C(CC)C)ccc(=NC(=O)C23CC(CN2C(=O)C(C)(C)C(C)(C)C)C3)[nH]1 61231,Cc1noc(C)c1CN(C(=O)C(C)SC(C)C)C.c12cn(C)nc1C2 61232,Cc1conc1C1CN(C(=O)CCCCC2C(CC(=O)NC(=O)C(C)C)C2)C1 61233,C1(CNC(Cc2ccc(C)cc2)=O)CCN(C(c2cc(Cl)ncc2N)=O)CC1C 61234,C1(C(N2CC(N(C)C)C2)=O)CCC2(CCCCC2)N1 61235,C1(C(N2CC3C(NC(C4N(C)C(=O)CC4)=O)(CC3)C2)=O)CC(C)(C)SC(C)(C)C1 61236,c1(OC)cc(C(=O)O)c(CNC2=NC(C)CS2)cn1 61237,c1(NS(CCC)(=O)=O)cccc(C(=O)NCCCNC(=O)CCN(C)CCO)c1 61238,CC1(C)CCN(C(c2cc(C3CC3)no2)=O)C(C(=O)NCC2(C)CCCO2)C1 61239,c1(C(=O)NCCOC2CN(C(C(N3CCC(C)C3)=O)=O)C2)c(F)cccc1F 61240,c1(C(N2CCCC(CN(C(=O)C(O)COC)CC)C2)=O)cnc2cc(C)ccn12 61241,C(C(C(=O)NCc1cnco1)NC(c1ccnnc1)=O)OCC 61242,C1(NC(C2(CCCC)CC2)=O)C=CCC(C(=O)NCCNc2nccs2)C1 61243,N1(C(C(=O)N(CCCNC(=O)NCC)CC)=O)CCOC(CSC)C1 61244,C=CC1(C(=O)NC(c2ccncc2)C)CCN(C(c2cnsc2C)=O)C1 61245,C(=O)(C(CCSc1ccccc1)OC)NCCN(C(=O)CCC1(C)CC1)CCC 61246,N1(C(c2n(CCC)ccc2)=O)CC(NC(=O)Cc2cnn(CC)c2)C(C)C1 61247,c1(C(N(CC(C)NC(c2nocc2Br)=O)C)=O)cccc(Cl)n1 61248,c1(CC)nc(C)n(C)c1C(=O)NC1C2CN(C(c3csnn3)=O)CC12 61249,C(=O)(CCC(=O)c1cccnc1)N1CC(CCCC(=O)O)(OC)C1 61250,c1(CC(CNC(C(c2cn(C)nc2)O)=O)CCO)c[nH]c2cccc(Br)c12 61251,C1(O)(CN(C)C(c2cc(Cl)cc(Cl)c2)=O)CCN(C(c2cn(C)nn2)=O)CC1 61252,c1(CC)cc(Cl)ccc1C(=O)NC(CN(C)C(C1CCOC1CC)=O)(CO)CO 61253,Cc1cc(C(N2CCCC3(C(=O)OC(C)(C)C)CC23)=O)cnc1-n1cccn1 61254,C1(C#N)(CC)CN(C(=O)C=CC2CCCN2C(=O)Cc2ccnc(O)c2)C1 61255,N1(C(Cc2c(C)nsc2)=O)CCN(C(=O)C(C)NC(N)=O)CC(C)(C)C1 61256,C1(O)(CN(C(C2C(OC)CCC2)=O)C)CCCN(C(c2ccncc2Cl)=O)C1 61257,C#CC1(C(N2CC3CCC2C3)=O)CN(C(=O)CCc2ccc[nH]2)C1 61258,c1(NC(C(CC)OC)=O)cccc(CC(F)(F)F)c1.c12ncc(s1)c(=O)[nH]2 61259,c1(CNC(C2(C3N(C(CCC4(C)CC4)=O)CCC3)CC2)=O)cccc(C(F)F)n1 61260,C1(NC(C2SCCS2)=O)COC2(C1)CN(C(c1occc1Br)=O)C2 61261,C(=O)(CC(C)P(C)(C)=O)NCC12N(C(c3c(C)cns3)=O)C(CC1)CC2 61262,c1(C(=O)NC2CCCC(CNC(CC(C)(C)N(C)C)=O)C2)ccc2c[nH]nc2c1 61263,CC1CC2(CCO1)CCN(C(=O)Cc1ccc([N+](=O)[O-])cc1C(=O)O)C2 61264,C1(O)(C(C)CNC(=O)C=CC(F)(F)F)CCN(C(c2cnc(S)n2C2CC2)=O)C1 61265,N1(C(Cc2cc(C(N3C4CCC3CC(O)C4)=O)no2)=O)CC(=O)N2CCCC2C1 61266,CCC(CC)CC(=O)NC1CC(CNC(c2ccc(C)nc2N)=O)C1 61267,C1(C2CCCCC2)(C(=O)NC(CNC(C(COCC)(C)C)=O)C2CCC2)CC1 61268,c1(C(=O)NCCCN(C(CC(C)C2CCCC2)=O)C2CC2)nccc(C(F)F)n1 61269,C1(CCCNC(c2c(C)scn2)=O)CCCCN1C(=O)CCc1ccncc1 61270,C1(CNC(CN2CCC(N(C(CC)=O)CC)C2)=O)CCc2nn[nH]c2C1 61271,c1(C(=O)NC(CC)C(=O)NCC(O)CCO)cc(Cl)cn1C 61272,c1(C(=O)NC(C2(O)CCN(C(CC=CC)=O)C2)C)cc(F)cc2cc[nH]c12 61273,N1(C(C2CC2COCC)=O)CC2CC(NC(c3ccnn3C3CC3)=O)CC(C2)C1 61274,CC(C)C(C(=O)NC1CC2CCC1O2)SCc1ccccc1 61275,c1(C(N2CC(NC(C(C=CC)O)=O)CC2(C)C)=O)cc(S(=O)(=O)N(C)C)c[nH]1 61276,C1(CN(C(=O)CCOC2CCC2)C)CN(C(c2c[nH]c(C#N)c2)=O)CCO1 61277,C(c1ccccc1)=C(C)C(N1CCCC1CC(=O)NCc1[nH]cnc1C)=O 61278,C(CN=c1nc(N2CCC(C)C3(CCC3)C2)c2c([nH]1)COC2)N(CCO)CC 61279,C1(C(N(C(CC)CO)CC)=O)CCCC(NC(=O)CC2CC3C=CC2C3)C1 61280,c1(C(N2CCC(NC(C(C)NC(COC)=O)=O)C2CO)=O)cc(O)cc(N)c1Cl 61281,C(=O)(C(C)(C)C(F)c1ccccc1)N1CCC(NC(c2c(Cl)cn(C)n2)=O)C1 61282,c1(C(N2CC(C)C(Cc3ccccc3)C2)=O)cnc(O)n(C2CC2)c1=O 61283,c1(C(N(C(C)CCNC(=O)CC2CCOC2)C)=O)cc(Br)cc2nc[nH]c12 61284,CCC(O)CCc1cn(CC2CC(NCc3cnn(CC4CCOC4)c3)C2)nn1 61285,c1(C(=O)NC(C(C)NC(C(C)NC(COC)=O)=O)CO)ccc(CC2CC2)cc1 61286,CC(c1ccc(F)cc1)=CC(=O)N(CCCNC(c1ccc(CC(C)C)s1)=O)C 61287,N1(C(C(CCC)O)=O)CCN(C(C2CCC2CF)=O)C(c2ccncc2)C1 61288,c1(C(=O)NCC2N(C(C3CN(CC)C(=O)C3)=O)CC2)cc(OC)c(OC)cc1F 61289,C1(C(N(C)CCc2cccnc2)=O)CC(O)CN1C(=O)Cn1cc(Cl)cn1 61290,C1(NC(Cc2c(CC)con2)=O)CCC(NC(=O)COCC(F)(F)F)CC1 61291,c1(OC)ccc(F)c(F)c1C(N1CC(C)CC1C(N1CCC(C(N)=S)CC1)=O)=O 61292,Cc1ccc(C2CC2)c(C(N2CC(O)(C(C)NC(c3conc3C)=O)C2)=O)c1 61293,N1(C(C2(COC)CC2)=O)CCC2(CCN(C(=O)Cc3ccsc3)CC2)C(C)C1 61294,N1(C(C(C)N=[N+]=[N-])=O)Cc2[nH]nc(C(=O)Nc3cccc(N(C)C)c3)c2C1 61295,CCC(C)(C)COCC(=O)NC(c1cn(-c2ccsc2C(=O)O)nn1)C(=O)O 61296,CC(C)(CN=C(NC1CCOCC1)NCC1(C)CCCO1)Oc1ccccc1 61297,C(CC1C(=O)NCCC(=O)N1)SC.C(CC(C(C)C)N(C)C)NC(N)=O 61298,C1(C(N2CCC(N(C(c3cnc(S)nc3)=O)CC)C2)=O)NC(=O)OC1(C)C 61299,c1(C(C)(C)C)cc(C(=O)NC2CCC(CCNC(=O)Cn3cnnc3O)C2)on1 61300,N1(C(Cc2cccc(C)c2Cl)=O)CC2CC1CCN2C(c1nncn1C1CC1)=O 61301,C(=O)(C(CC(C)C)OC)N1CC(CCC)C(C(N2CC(CC(=O)OC)C2)=O)C1 61302,c1(C(N(CC(CN(C)C(c2c[nH]cc2C(F)(F)F)=O)O)C)=O)ccc(N)c(O)c1 61303,N1(C(CC(CCC)O)=O)CC2CCC1CN2C(=O)C(C)Cc1cccc(F)c1 61304,N1(C(Cc2cccc(C)c2)=O)CCC(C(=O)Nc2cnc(C#N)cn2)C(O)C1 61305,N1(C(=O)NC(c2csnn2)C)CC(COC(C)(C)C)C(O)C1 61306,N1(C(c2cc(COC)on2)C(=O)NC(CC)C)c2ccccc2CC1C 61307,c1(CC)ccc(CO)cc1.C12C(C1(F)F)CC(=O)N(C)CC1(CC1)CNC2=O 61308,c1(N(CCCN(C(=O)CCc2cc(C)no2)COC)CC)c(F)cccc1[N+](=O)[O-] 61309,CCCCCCC(CC)NC(C1CC=CCC1NC(c1cscn1)=O)=O 61310,CC1(NC(c2n[nH]c3c2COC3)=O)CCC(NC(C2(C)CCCCO2)=O)CC1 61311,C(C(C)(O)CC(C)C)NC(CC1C2CN(C(C(C3CCC3)OC)=O)CC21)=O 61312,CC12COCC1CN(C(=O)CCc1nnc(C3CCCC3)o1)C2 61313,CCC(=O)N(CCC(=O)NC1CCN(C)CC12CCC2)OC 61314,C(=O)(C1=NN(C)C(=O)CC1)NC1CCC(NC(c2c(C)c(N)cnc2)=O)C1 61315,n1(CC)cnc2c(N(CCS(C)(=O)=O)C)[nH]c(=NCCC(N)=O)nc12 61316,C1(C(=O)NC(CCOC)CNC(c2ccc(Cl)s2)=O)CC2(C1)NC(=O)NC2=O 61317,c1(C(N2C(CO)CC(C)C2)=O)ccc2c(-c3ccc([N+](=O)[O-])cc3F)n[nH]c2c1 61318,C1(NC(C=CCNC(C2CN(C(C)C)C2)=O)=O)(CO)CC2CCCC12 61319,C1(F)(CNC(C(C2CCCO2)OC)=O)CC(CNC(=O)COCC(F)F)C1 61320,C(C)(CCN=c1[nH]c(=NCC(C)(C)N(C)C)[nH]c2ccc(Cl)cc12)OC 61321,N1(C(c2c(Cl)ccnc2Cl)=O)CCC2C(CCN2C(=O)Cc2cccc(Cl)c2)C1 61322,C1(C)(CNC(C(C)S(C)(=O)=O)=O)CN(C(c2ncc3ccccn23)=O)C(C)(C)C1 61323,N1(C(CC=C=C)=O)CCC(C)(C)C1C(=O)NC1CC2OCCCC12 61324,N1(C(C(C)OC)=O)CC=C(CNC(c2ncccc2Cl)=O)CC1 61325,c1(CNC(C2CCC(CNC(=O)CCn3cnnn3)C2)=O)cnccc1Cl 61326,N1(C(CCc2ccc(C)o2)=O)CCC(CNC(c2ccnn2C(F)F)=O)C(C)C1 61327,Cc1cccc(C(=O)N(CCCNC(=O)C(c2cnccn2)C)C2CC2)c1Cl 61328,c1(CC(=O)NC2CC(NC(Cc3c(C)n[nH]c3C)=O)C2)c(F)cccc1Br 61329,C(=O)(CCCC(F)(F)C(F)(F)F)NC1CN(C(C(COC)N(C)C)=O)CC12CC2 61330,N1(CCN(C(CC2C(C)CCC2)=O)C(C)C)CCN(C(=O)C(C)(C)N(C)C)CC1 61331,c1(C(=O)NCCCNC(N(C(C)C)C)=O)cccc(Br)c1 61332,C(=O)(CC(C(C)C)NC(c1cnncc1C)=O)N1CCC(CC)(CC)C1 61333,c1(C(N2CC(OCC)(CNC(C3C=CCCC3)=O)C2)=O)c(CC)nn(C)c1Cl 61334,N(C1CCc2cccc(Cl)c21)c1c(C)c(NCCCC2CCCCC2O)ncn1 61335,c1(C(=O)NC(CNC(c2cnc(OC)s2)=O)C)sc(F)cc1Cl 61336,C1(CC)CC(OC)CN(C(C)C(=O)NCCOC(c2ccccc2)C2CC2)C1 61337,N1(C(c2nccc(OC)c2OC)=O)CCC(NC(C2CCC2)=O)C(C)(C)C1 61338,N1(C(c2cnn(C(C)C)c2Cl)=O)CCN(C(=O)CCc2cc[nH]n2)CC1C(F)F 61339,c1(C(N(CC(C)NC(C(C2CCOCC2)OCC)=O)C)=O)[nH]cnc1C#N 61340,N1(C(c2c(C)nsc2C)=O)C2CCC1C(C)C(NC(C1CC(C)(C)CN1C)=O)C2 61341,N1(C(c2n(C)c(Cl)nc2)C(=O)NC2CC2)CCN(Cc2ccccc2Cl)C(=O)C1 61342,C1(N(C2CCC(C(=O)OC)C2)C(c2nnc(C)n2C)C(=O)OC)CC2CCC1C2 61343,c1(NC(N2CCN(C3CCOC34CCOC4)CC2)=O)c[nH]c2cccnc12 61344,c1(C(N2CCC(CCNC(c3csc(S)n3)=O)CC2)=O)cccc([N+](=O)[O-])c1 61345,N1(C(C(CC#C)CC#C)=O)CC2CCCC(C1)N2C(=O)CC1(C(F)F)CC1 61346,Cc1cc(=NC(=O)c2ncccc2-n2cccn2)[nH]n1CCSC1CCCCC1 61347,C1(OC(C)C(N2CC(O)(CCNC(C3(C#N)CCC3)=O)C2)=O)CCOCC1 61348,CC(C)CC(C)C(=O)NCC1CCCN(C(C2CCCN2c2ncccn2)=O)C1 61349,C1(NC(c2nn(CC)nc2C)=O)CCN(C(=O)CCc2cscn2)C12CCC2 61350,n1(CC(=O)NCC(CNC(C2(Cl)CC2(C)C)=O)OC)cc(C)cn1 61351,c1(OCCCC(N2CC(NCCOC)OCC2)=O)cc(C)ccc1C 61352,c1(C(N2CC3CCN(C(CC(C)SC)=O)C3C2)=O)ccnc2ncccc12 61353,C1(NC(c2ccc(CCF)cc2)=O)CCC2CN(C(C3CCCO3)=O)CC2C1 61354,c1(OC)cc(C(N2CCCC2C=CC(=O)NCC2CC2(C)C)=O)ncn1 61355,C(N=c1[nH]nc(COC)s1)C1CN(C(CC2(OC)CC2)=O)CC1C(F)(F)F 61356,CCC(CCC(=O)Nc1ccc(C(C)C)nc1)NC(=O)C(C)c1cccs1 61357,C1(C(=O)N(C)CCN(C)C(C2CC=CCC2)=O)(NC(C)=O)CCC(C)CC1 61358,c1(C(=O)NC2CC(NC(C3CCC(CN(C)C)O3)=O)C2)n[nH]c2c1CN(C)CC2 61359,CCCC(C)(O)C(=O)N1CCOCC(NC(=O)C(C(C)C)c2ccccc2)C1 61360,C1(NC(c2cnn(C3CC3)c2)=O)CC2CCC1N(C(c1ccsc1)=O)C2 61361,CC(C)C(CC(=O)NC1(C)CCN(C(c2cc(C#N)on2)=O)C1)c1ccon1 61362,c1(C(N2CC(C)C(NC(=O)C=CCN(C)C)CC2)=O)ccc2c(c1)C(=O)NCC2 61363,C1(C(N2CC(NC(C=Cc3ccn(C)c3)=O)(CO)C2)=O)CCc2ccnn2C1 61364,C1(C(=O)NCc2nnc(C)o2)(CF)CCN(C(=O)COC2CCOC2)C1 61365,C1(CCNC(C(CO)OC)=O)CCN(C(C2C3COCC23)=O)CC1(F)F 61366,CC1CC(C(=O)NCCN2CCN(CC(F)(F)F)CC2)CCS1 61367,C1(C(N(CC(=O)O)Cc2cn(C3C(C)(O)CCC3)nn2)=O)CC2(CC(=O)C2)C1 61368,C(C(C)(C)C(=O)NC(CNC(c1cc(Br)oc1C)=O)C(C)C)NC(C)=O 61369,N1(C(c2nc(C(C)OC)sc2)=O)CCC2CCN(C(c3cc(N)ccn3)=O)CC12 61370,Cc1cc(NC(C2(C)CN(C(=O)CCc3ccccn3)C2)=O)cnc1F 61371,c1(C(=O)NC2C(C(=O)NCC(c3cccc(O)c3)O)CCC2)cccc(F)c1F 61372,C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CN(C(=O)C=Cc1ccccc1Cl)C)(C)C 61373,C(=O)(C1CNC(=O)c2ccccc21)Nc1ccc(C)c(I)c1 61374,N(C(=NCC1CC1(F)F)NCC1CCCO1)C1CC(OCC(=O)NC(C)=O)C1 61375,N1(C(=O)NCCCCC(OC)NC(=O)OCCN=[N+]=[N-])CC2(C1)OC(=O)NC2C 61376,C1(NC(C2(C(N)=O)CC2)=O)CC(CNC(=O)C=CC2CCCO2)C(O)C1 61377,N1(CC(CCC=C(C)C)C)CC(O)CC12CCS(=O)(=O)CC2 61378,Cc1oc(C(N2CCCCC2CNC(c2ccc(C(C)(C)C)[nH]2)=O)=O)cc1Br 61379,Cc1cnc(C(N2CC3CC2C3CNC(=O)C(C)Cc2ccccc2)=O)nc1 61380,N1(C(C(F)=CCC)=O)CCN(C(C2CCCCC2(C)C)=O)CC1CS(C)(=O)=O 61381,c1(SCC(=O)NC(CC)(C)CNC(=O)Cn2nnc(C3CC3)n2)ccnc(Cl)c1 61382,C(=O)(C1=C(Cl)CCC(C)C1)NCC(CCCC)NC(c1ccc(Cl)o1)=O 61383,c1(CNC(c2c(C)coc2C)=O)cc(O)nc(CNC(=O)CC(O)C(C)C)n1 61384,c1(OC)ccc(-c2ccc(N)cc2CNC)cc1COC1CC(C)C1 61385,C(C(F)(F)C(=O)NCC1(NC(=O)C(n2cc(C)cn2)C)CCCCC1)OC 61386,CC(C)CC(CNC(=O)C(C)C(F)(F)F)C(=O)Nc1ccc2nc[nH]c2c1 61387,CCC(C)(C(=O)NCC1(F)CCN(C(C2(C)COCCO2)=O)CC1)C(F)F 61388,c1(OC)cc[n+]([O-])c(C(=O)NCC(O)CCNC(=O)C2=NNC(=O)C2)c1 61389,N1(C(Cc2ccc(C)c(C(N3CCCC3)=O)c2)=O)CC(C(=O)O)CCC1(C)C 61390,C(=O)(CC1=Cc2ccccc2C1)N1CC(OCC)C(CNC(C2CC2C)=O)C1 61391,C=C(C)CCCC(=O)N(C(CNC(c1ccc(OCCC)c(N)c1)=O)C1CC1)C 61392,C#Cc1ccc(C(N2CC(C3(NC(=O)C(CC4CCCC4)CC)CC3)C2)=O)cn1 61393,N1(C(C2=C(C)OCCS2)=O)CC(NC(=O)C(C)c2cncs2)CC2(CCC2)C1 61394,Cc1cn2cc(C(=O)NCCC3(O)CN(C(C4(O)CCOCC4)=O)C3)sc2n1 61395,N1(C(=O)NC(c2cnccn2)C2CC2)CC2CCC(CO)(C2)C1 61396,N1(C(C(CC)OC)=O)CCC(CC(N)=O)(NC(=O)CC(CC)SC)CC1 61397,N1(C(C2C(C(C)C)C2)=O)CCC2CN(C(c3cn(CC4CCOC4)nn3)=O)C2C1 61398,C#Cc1nc(C(N2CCN(C3CCC(NC(=O)CS(=O)(=O)NC)C3)CC2)=O)cs1 61399,C(=O)(C1=CCC(C)(C)CC1)NCC1CCN(C(COC(CC)C)=O)C1(C)C 61400,C1(NC(C(C(C)C)C#N)=O)CN(C(C2CC3(CSC3)C2)=O)CC2(CCC2)C1 61401,c1(N(C(C(CC)C)=O)C(Cc2ccc(F)cc2)C(=O)O)ncc(OC)cn1 61402,C(C)(C(O)C(=O)NCC1(CCNC(=O)CCn2nc(C)cc2C)CC1)SC 61403,C(CCCCCNC(=O)OC(C)(C)C)NC(N(C)C)=O.c1(C(C)O)ccoc1C 61404,C(=O)(C(Cc1ccoc1)NC(=O)CCC1(C)N=N1)NCC(C)F 61405,C1(CNC(c2c(COC)cco2)=O)CC2CCC1N2C(c1cc(OC)ns1)=O 61406,N1(C(CCNC(=O)NC)=O)CCN(CCNC(C2CC2CF)=O)CC1 61407,N1(C(C(C)SC(C)C)=O)CCC(C(O)CNC(=O)C(C)n2cncn2)CC1 61408,c1(-c2cnc(NC(Cc3ccc(C#N)cc3)=O)c(C)c2)cnc2ccc(F)cc2c1 61409,CC(C)CC(O)C(=O)NCC(Cc1ccccc1)NC(C1CC1(Cl)Cl)=O 61410,C1(CNC(C(C)CO)=O)CC2CC2N1C(c1cccc(C2CCCC2)c1)=O 61411,N1(C(C(CO)N(C)C)=O)CCCCC1CNC(c1ccc(-c2ccncc2)s1)=O 61412,c1(OC)ccnc(F)c1C(=O)NCC12CC(CN1C(=O)C(C)OC)C2 61413,C1(n2cc(CCOC(C)=O)nn2)CCCN(C(c2csc(C(F)F)c2)=O)C1 61414,c1(C(=O)NCC2CN(C(c3c(Cl)nc(OC)s3)=O)CC2C)cc2ncccn2n1 61415,Cc1ccc(C(N2CCCC(NC(C3(C4CCCO4)CC3)=O)C2)=O)c(F)c1C 61416,c1(C(=O)NC(CCCN(C(=O)C(N)=O)C)(C)C)ccc(N=c2cc[nH]cc2)cc1 61417,Cc1cc2c(C(=O)NCCCCCCN(C)C(C3CCCC3O)=O)cccc2[nH]1 61418,C(CN=c1[nH]c(=NCCN2CC3CCCC3C2)[nH]c2c1COC2)n1c(=O)cccc1 61419,CCC(C)(C)C(=O)N1CCC(C(=O)NCCN=[N+]=[N-])O1 61420,C#CCCC(O)C(=O)NCC(C)CNC(=O)CCC(=O)NC(c1ccccc1)C 61421,CC(C)C(C(=O)OCC(=O)NC(c1nncs1)C)n1cc(Br)cn1 61422,Cc1ccc(C(=O)NCC(C)(C)C(N2CCCC(CO)C2C)=O)cc1C 61423,C1(CC(N2CCC(n3cc(C(C)NC)nn3)CC2)=O)CC2CCC1NC2 61424,Cc1nc(CC(N2CC(OCCNC(c3cc(CO)[nH]n3)=O)C2)=O)co1 61425,CCC(C)(C(=O)NCCC1CC(NC(C2CC2c2cccnc2)=O)C1)C(F)F 61426,CC(C)CC(F)(F)C(=O)NC1CCCCC1CNC(=O)CCC1CCCCN1C 61427,n1(CC=C)nnnc1C(c1c[nH]nc1CCC)NCCCc1nnc(C)s1 61428,c1(C(=O)NC2CCCC(NC(C(COC)(F)F)=O)C2)cccc2c1NC(=O)CC2 61429,C1(NCCC2CC(OCC)C2)CCS(=O)C1 61430,c1(C(=O)NC(C(C)(C)NC(C(COCC)C)=O)C)cc(C)n(C(C)C)n1 61431,Cc1c(C(=O)NCC(C)CN(C(=O)C=C2CCC(C)C2)C)ncn1C 61432,C(=O)(CCC(=O)NC1CCCCC1CNC(=O)CCCN1C(=O)CCC1=O)NC 61433,C1(C(=O)NCCCCCCC)CC2(CCN1C(C1CN(C(C)=O)C1)=O)CC2 61434,C1(NC(c2c(CC)scc2)=O)CCC2(CCCN(C(=O)CCC(CF)CF)C2)C1 61435,Cc1nc(C)c(S(=O)(=O)NC(C(C)C)C2(CO)CCC2)o1 61436,C1(C(=O)Nc2ccc(C#C)nc2)CCN(C(=O)CC(CN(C)C)CC)C(C)(C)C1 61437,N1(C(c2cc3sccc3[nH]2)=O)CC2CCN(C(=O)CC34CCC(CC3)C4)C2C1 61438,c1(C(=O)NC(C)CN(C)C(c2n[nH]c(C3CC3)n2)=O)cc(Cl)c(Cl)cc1N 61439,C1(C(N)=O)CCCC(NC(=O)CC(CC2CC2)NC(c2cn(CCO)nn2)=O)C1 61440,C(CCCCCNC(=O)C(F)n1ccnc1)NC(=O)CCCn1ccnc1 61441,C12(C(=O)NCCCN(C(=O)CCOC(C)CC(C)C)CC)CCCC(CO1)C2 61442,Cc1nc(C#N)c(NCCC(=O)NCC2CN(C(C3CCSC3)=O)C(C)(C)C2)o1 61443,C1(CC2CC(NC(N(CC(N3CCCC3)C)CC#C)=O)C2)CCC(=O)N1 61444,c1(C(N(CC)CC2CCCN2C(C2CCC2)=O)=O)ccc2cccc(F)c2n1 61445,O=S1(=O)CC(CNC(=NCCc2ccns2)NCC2CCC2)Oc2ccccc21 61446,CC(C(=O)N1CC(O)CC1CNC(c1ccc(CCN(C)C)cc1)=O)C(C)(C)C 61447,c1(C(=O)NCCC(C)CCNC(C2CCCOC2C)=O)ccc2c(c1)C(=O)NC2 61448,Cc1ncc(C(=O)NC(C2(CNC(=O)CCN3CCCCC3C)CC2)C)c(=N)[nH]1 61449,CCC(CC)CCC(=O)N1CC2CC1CC2NC(c1sc(C)nc1C)=O 61450,N1(C(=O)CCN(CCO)CCO)CC=CC1Cn1cc(C(C2CC2)N(C)C)nn1 61451,c1(OC)nc(C(=O)NCC2CC3CC3N2C(=O)C=CC(C)C)cc(O)n1 61452,C(=O)(C1=C(Cl)CCOC1)N1CCC(N(C(=O)CSCc2ccccc2)C)CC1 61453,C1(NC(c2ccc(Cl)cn2)=O)CCN(C(c2cccc(C(F)(F)F)c2)=O)CC1F 61454,N1(C(c2cnc(C)[nH]2)=O)CC(NC(c2cc(C(C)(C)C)nn2C)=O)C(C)C1 61455,C(=O)(N1CC(O)CCO1)c1cc(CNC(C(=CC2CCCC2)C)=O)nn1C 61456,N1(C(CCCCC)=O)CCN(C(CC(C23C4C5C6C4C2C6C35)=O)=O)CC2(CC2)C1 61457,C1(C(=O)NCc2cscn2)CC12CCN(C(c1cnc(Cl)cc1Cl)=O)C2 61458,C1(NC(CC(C)OCc2ccccc2)=O)CN(C(=O)C(Cl)=CCl)CCC1(C)C 61459,N1(C(CC2(OC)CCC2)=O)CC2CC1CN2C(=O)CCC(C)n1cccn1 61460,C(CCC(CC)CC)NC(=NCC=C)NCC(C)(C)C(=O)OC 61461,N(C(=NCC(F)(F)Cl)NCC(=O)N(C)Cc1ccccc1)C1CCC(OC)CC1 61462,C1(N(C(C=CC)=O)C)CCCN(C(=O)NC2CC2c2ccncc2F)C1 61463,c1(C(=O)NCC2C(NC(c3cc(C)sc3C)=O)COC2)cnc2ccoc2c1 61464,N1(CC)CCC(CNC(C2C(C)CCN2C(C2CC(F)CN2C)=O)=O)CC1 61465,c1(C2(C)CC2)ccccc1NC(=O)C=CCNC(=O)CC1COCCOC1 61466,N1(C(=O)Cc2cc(C3CC3)on2)CC2CN(C(C3(F)CCC3)=O)CCC12 61467,c1(C(N2CCC(NC(CN(c3ccncc3)C)=O)C2)=O)ccnc(Cl)c1O 61468,c1(C(N2CCC(Cn3cc(CC)nn3)C2)=O)c[nH]c2c(C)c(Cl)ccc2c1=O 61469,c1(C(N(C(C)CNC(=O)CSCC(F)(F)F)C)=O)csc(C(F)(F)F)n1 61470,C1(C(N2CCC(NC(c3c(C(C)(C)C)con3)=O)C2)=O)CC2(C1)CC(F)C2 61471,C(c1cnn(C)c1C)=CC(=O)NCCN(CCC)C(c1cc(OC)ccc1Cl)=O 61472,n1(CC(=O)NCCC2=CCN(C(=O)C=C(Cl)Cl)CC2)nc2n(c1=O)CCCC2 61473,CC1CCCCCN1C(c1ccoc1CNC(C1COCC1(C)C)=O)=O 61474,C=CCC(C(=O)OCC)NC(=O)CC1C=CC(NC(=O)C(C)C=C)C1 61475,c1(C(=O)NC(C2CN(C(CCNC(C)=O)=O)C2)C)ccnc(S)c1 61476,C1(CCC)CN(C(c2sccc2F)=O)CC1NC(=O)CN(CC)CC 61477,CCC(C(=O)NC1(C)CCC(NC2(CC(=O)NC3CC3)CC2)CC1)C(C)(C)CC 61478,N1(C(CCCC(N)=O)=O)C2CCCC1CN(C(=O)CCOC1CC1)CC2 61479,Cc1cc(CNC(N2CCC(C)CC2C(C)O)=O)cnc1C 61480,C(=O)(C(C)(O)CC(C)C)N1CC(N(C(c2[nH]cc(C)c2)=O)C)C(C)(C)C1 61481,N1(C(CCC2CCC(NC(=O)C(c3ccccc3)O)C2)=O)CCCCCC1CO 61482,c1(C(N(CC(C)NC(=O)Cn2cnc(=N)[nH]2)CC)=O)ccc(C(C)F)cc1 61483,C1(C2CCOCC2)(C(N2C(CNC(C=C(CC)CC)=O)CC2)=O)CC1 61484,n1(CC(=O)N(C(C)C(=O)NC(CC)C(C)O)CCC)ccc(C)n1 61485,Cc1nsc(C)c1NC(C1(NC(=O)CC(=O)N(C)C)CC(F)C1)=O 61486,N1(C(C2CC(C)(F)C2)=O)CCC2C(C1)NC(=O)CN2C(c1ccc(O)c(Cl)n1)=O 61487,c1(C(=O)NCC(CO)NC(c2c(C)nco2)=O)cnc(S)nc1 61488,C1(CC(N2CC(NC(c3ccc(OC)s3)=O)C(C(F)F)C2)=O)C(=O)N(C)N=C1C 61489,C1(C(=O)NC(CCNC(c2c(CC=C)cccc2)=O)(C)C)CS(=O)(=O)CCO1 61490,N1(C(CC2(COC)CC2)=O)C(C)CN(C(=O)C#CC(C)(C)O)CC1C 61491,CC1(CNC(=O)C=Cc2ccccc2)CCC(NC(=O)CNC(=O)C(C)(C)C)CC1 61492,N1(C(c2c(NCC)ccc(Cl)c2)=O)CCC(C)(C)C(NC(=O)CCC2CC2C)C1 61493,N1(C(CCC)=O)CC2CCC(NC(=O)CCC(C)c3ccccc3)CC2C1 61494,C1(NC(C2CCCN(CC)C2)=O)CCN(C(C2CC(C)C2)=O)CCC1CO 61495,N1(C(c2c(CC)nns2)=O)CCC(NC(c2nccnc2C)=O)C(CO)C1 61496,c1(C(=O)NCCC2(O)CN(C(C(C)=O)=O)C2)ccc2c(c1)CCC=C2 61497,C(=O)(C1COc2c(F)cccc21)Nc1ccc(C)c2c1CCCC2 61498,N1(C(CCOCC)=O)CC2CC(NC(=O)C(C)OCC(F)(F)F)CC1C2 61499,CC(C)(C)CCCCNC(C1C(CNC(=O)CCc2ccccn2)C1(C)C)=O 61500,C(=O)(C(O)P(C)(C)=O)N1CC(c2cn(C)nn2)C1.C1(COC)CCCC1 61501,Cc1c(C(N2CC3CCC3(CC(N3CCOC(C(N)=O)C3)=O)C2)=O)[nH]ccc1=O 61502,c1(OCCNC(=O)NCc2cncc3c2CCCC3)ccc2ccccc2c1Br 61503,c1(C(=O)NCCN(C(c2cn(CC)nn2)=O)C(C)C)c(F)cc(Br)c(F)c1F 61504,NS(=O)(=O)C1(C(=O)NCCN(C2CCCCC2)C(C2CC(F)(F)CS2)=O)CC1 61505,C(=O)(C(F)C(C)(C)O)NC(CC=C)CNC(c1cnn(-c2ccc(F)cc2)c1)=O 61506,CC(CCCCNC(C1CCC(=O)N1C)=O)NC(c1ccn(CCF)n1)=O 61507,c1(C(N2CCOC(c3ccco3)C2)C(=O)NCC=C)ccc2cc(Br)ccc2c1 61508,Cc1cccn(CC(=O)NC2CC(F)CN(C(=O)Cc3ccc(Cl)nc3)C2)c1=O 61509,N1(C(=O)C(C2CC2)NC(C23CSCC2C3)=O)CC2(CCOC2)C1 61510,C(=O)(CCCCC(=O)NCCC1(O)CCN(C(=O)CCCc2nccs2)C1)NC 61511,C12(C(=O)NCC(C(C)C)NC(=O)COCC3CCCCO3)CCCC(C)(C1)OC2 61512,Cc1cc(=NCCCCC#N)[nH]cc1S(=O)(=O)N1CCC(C)C1C 61513,c1(NC(c2n(CCOCC)nnn2)c2scnc2Br)ccc2cnn(C)c2c1 61514,c1(C(N2CCC(CC)C2CNC(c2cncc(OC)n2)=O)=O)nc(C)ccc1C 61515,CC1(C)COC(CCNC(=O)C=Cc2ccc(Br)o2)C1 61516,c1(C(C)C)nc(C(=O)NCCN(C(C2CC3CC3C2)=O)CC2CC2)cs1 61517,N1(C(CCNS(CC)(=O)=O)=O)CCC(NC(=O)CSC(=N)N)C(F)C1 61518,N1(C(C2C(C=C)CC2)=O)CCc2nc(CNC(C3(C)CC(C)=NO3)=O)sc2C1 61519,C(=O)(C(C)(C)CS(C)(=O)=O)NC1C(C(=O)Nc2c(C)ncn2O)OCC1.C1(C)CO1 61520,N1(C(C(CCC)OCC)=O)CCC(C2CC2)C1C(=O)NC1CCCC1CN(C)C 61521,C1(C(N(CCC)C(c2cccc(-c3nn[nH]n3)c2)C)=O)CC2CCC1O2 61522,C1(NC(c2cc3sccc3[nH]2)=O)CC2CN(C(C3SCCCS3)=O)CCN2C1=O 61523,C1(C(=O)OC)CN(C(C2CC(C)N(C(=O)OC(C)(C)C)C2)=O)C(C)(C)C1 61524,N1(C(CCC=CCC=C)=O)CCC(C(=O)NCCS(=O)(=O)NC)C1CC 61525,N1(C(Cc2c(C)occ2)=O)CCOCC1CCNC(C12CC(C(F)F)(CO1)C2)=O 61526,C1(CNC(c2cnn(CC)n2)=O)CC(C)N(C(=O)CCCN(C)C(C)=O)C1 61527,C1(C(=O)NCC2(CCNC(c3nsnc3O)=O)CC2)(CC2CCC2)CCCC1 61528,c1(CNC(=O)C(c2ccccc2)Nc2ccccc2)ccc(S(F)(F)(F)(F)F)cc1 61529,N1(C(C(CC)(CC)CO)=O)CCC2(CCC2NC(c2cnc[nH]2)=O)CC1 61530,c1(C(C)NC(=O)CCn2cc(-c3cccc(CO)c3)nn2)cccc([N+](=O)[O-])c1 61531,C12(C(=O)NOCCC3CC3)CCC(CC1)N(C(c1cccc3[nH]ncc13)=O)C2 61532,C1(C(=O)NC(CC)C(=O)NC2CNC(=O)C23CC3)CC(C)(C)CCO1 61533,C(=O)(C(C)(C)S(C)(=O)=O)NC1C(c2n(C)ncc2)CN(C(C2CCOC2)=O)C1 61534,CC(C)(C)C(O)C(=O)NC1CC(F)CN(C(c2ccc(-n3cccc3)cc2)=O)C1 61535,C(=O)(C1=CCCC1C)NCC1(CNC(c2cc(C)sc2C)=O)CC1 61536,c1(C(=O)NCc2cnc(CC)[nH]2)cc(Cl)cc(Cl)c1F 61537,C(=O)(CCCCN(C(=O)C(C1CC1)OC)C)NC(c1cccnc1)CC 61538,N1(C(c2cc(CC)ncn2)=O)CCCN(C(=O)C=CCF)C(C(C)C)C1 61539,Cc1cc(F)c(N)cc1C(=O)NCC(CC(C)C)NC(=O)CC=C(Cl)Cl 61540,N1(C(C(CC#C)NC(=O)CN2CCCC2)=O)CCC(C2CC2)C1 61541,c1(OC)cccc(F)c1CNC(C1CCN1C(c1ccc(Br)s1)=O)=O 61542,c1(OC)ccccc1CNc1ncnc(NCCOC)n1 61543,N(C1c2ccccc2CC1(C)C)c1[nH]c(=NC23C(C)(C)C(CC2)CC3)[nH]c(=N)n1 61544,C#CCCCC(=O)NCCCC(C)NC(=O)C(O)Cc1[nH]cnc1C 61545,N1(C(c2ccc(CC)c(N)c2)=O)CC2CCN(C(c3ccc(CO)nc3)=O)CC12 61546,N1(C(C(CC)(COC)CC)=O)CC2(C=C(C(=O)NCCC(C)(C)OC)CO2)C1 61547,C(N=c1nc(N2CCC(CCO)C2)cc(C)[nH]1)C1(CCC=C)CCCC1 61548,C1(CNC(c2c(C)n[nH]c2C)=O)CC2(CC2)CN1C(=O)C=CCF 61549,CCCCCC(F)C(=O)N1CCC=CC1C(=O)N(CC1CCCCC1)OC 61550,C1(N(C(C(C)=CC)=O)C)CS(=O)(=O)C12CCN(C(C1(CO)CCCO1)=O)CC2 61551,C12(C(=O)OC)CNCC1(C(=O)N(C(C)C(N)=O)C(C)=O)C2 61552,c1(C(=O)NC2CC(C)(NC(C3CCOCC3)=O)C2)cccc2c1CCC2=O 61553,c1(C(=O)NCCN(C(=O)C(C)OC)CCC)cc2occ(Br)c2[nH]1 61554,C1(Nc2nc(C)nc(C#N)c2)CCC2(CC1)CN(C(C1CC1(C)Br)=O)CCO2 61555,c1(C(N(CC(O)CN(C)C(c2cc(O)ncn2)=O)C)=O)cc2c(=O)cc[nH]c2s1 61556,n1(CC(=O)N(C)CC2CCN(C(C3C=CCC3)=O)C2)cc(Br)c(O)nc1=O 61557,C1(c2n(CCCSCC)nnn2)(NCc2nnn(C(C)(C)C)n2)CC2CCCC12 61558,C(=O)(C1=NOC2(CCC2)C1)NC(C1(CNC(C2(C)COC(C)(C)CO2)=O)CC1)C 61559,C(=O)(CCCCC(N)=O)NC(C1CCCN1C(c1cc(CN(C)C)c[nH]1)=O)C 61560,N1(C(C(C)(C)N(C)C)=O)CCC(NC(C2CN3CCN2CC3)=O)C(O)C1 61561,N1(C(C(C)O)=O)CCN(C(=O)CCc2n[nH]c(=N)s2)C(C(F)F)C1 61562,CC(C)CC(C)(O)C(=O)NC(CNC(c1ccccc1SC(F)(F)F)=O)C(C)C 61563,C1(C(C)NC(COC(C)C)=O)CCN(C(=O)Cc2cnn(C)c2)CC1 61564,C(C)(CNC(=O)Cc1ccc(C)cn1)(CC(C)C)NC(C(C)OCC=C)=O 61565,Cc1c(C(=O)NC2(C)CN(C(=O)CC3CC4CCC3C4)C2)cncc1Cl 61566,C12(C(N3CC(CNC(C4C(CC)C4)=O)C(O)C3)=O)CCC(C(F)F)(CC1)C2 61567,C(CN=c1[nH]c(C)cc(=NCCCCO)[nH]1)c1c(SCC)ccc(OC)c1 61568,C1(NC(CCc2c(OC)cccc2)=O)CCN(C(=O)Cc2ncoc2C)C12CC2 61569,C=CCC(CNC(=O)CCCF)C(=O)N(C)CCn1cccn1 61570,Cc1cc(C(=O)NC2CCN(C(c3[nH]nnc3C)=O)C(C)C2)c2c(C)noc2n1 61571,N1(C(CC(C)C2CC2)=O)CCCCC1CCC(C)(C)NC(=O)CC1(O)CCC1 61572,N1(C(C2(C)CCN(C)C2=O)=O)CC2CCC1C(CNC(=O)C=Cc1ccoc1)C2 61573,c1(C(=O)NCC2C3CN(C(CCC)=O)C2C3)cc(Cl)c(Cl)c(Cl)c1 61574,C(CN=C(NCc1ncccc1C)N1CCC(F)(c2ccccc2F)C1)OC 61575,c1(C(NOCC(=O)NCC2(CC3CC3)CC2)=O)ccncc1F 61576,C(c1nc(C)c(C)[nH]1)=CC(=O)NCC(CC)N(C(C=CCCC)=O)C 61577,N1(C(CCC)=O)CCCN(C(c2cccc(N3CC=CC3)c2)=O)CC1CO 61578,n1(C2CC(C(N(CC=C)C)=O)C2)cc(-c2ncoc2C)nn1 61579,c1(C(N2CC(CCNC(CCC(=C)Cl)=O)(OC)C2)=O)coc2ccc(Cl)cc12 61580,N1(C(c2nc(OC)c(Br)cc2)=O)CC2CN(C(=O)C(O)C3CC3)CC2C1 61581,C(=O)(C(O)CC(F)(F)F)NC1CC(C(=O)NC(C2CCCCC2)C#C)C1(C)C 61582,C(C1=CCN(C(C2(C(F)(F)F)CCCC2)=O)CC1)NC(C1C(C)(Br)C1)=O 61583,n1(CC)nccc1C(=O)NC1(c2ccncc2)CCC1 61584,n1(CC(=O)NC(CNC(C(C)Oc2ccc(C)cc2)=O)C)c([N+](=O)[O-])cnc1C 61585,C1(CNC(C(CCC)C)=O)CC2(CC2)CN1C(c1cnc(O)c(Br)c1)=O 61586,C1(C(=O)NC2CC(CNC(c3cnn(CCF)c3)=O)C2)C2CC3C(C2)C13 61587,c1(CC)ccc([N+](=O)[O-])[nH]1.C12CCN(C1)C(=O)C1CCCN1N(C(C)C)C2=O 61588,c1(CN2C(CC(=O)Nc3ncc(C)c(F)c3)CCC2)ccc(Br)c2nsnc12 61589,c1(CCCC)ccc(C(=O)NC(C)C(C#N)CC)cc1C(F)(F)F 61590,c1(C(N2CCC(N(C(C3(CC)CCNC3=O)=O)C)CC2)=O)cc(O)cc(F)c1F 61591,c1(C(N2CC(NC(c3ncc(C)cn3)=O)C(C)CC2)=O)cccc2scnc12 61592,C1(CC)CN(C(=O)CC2COCC2(C)C)CCC1NC(C1CCCC(=O)C1)=O 61593,Cc1nc2c(NCC3CC(CNC(=O)Cn4ccnn4)CO3)ncnc2s1 61594,Cc1c(C(N2CC(CNC(c3c(F)ccc(F)c3O)=O)C2)=O)nn2c1OCCC2 61595,C(=O)(CCCC(C)(C)CC)NC1CN(C(c2c(CC)noc2)=O)CC1C(F)(F)F 61596,c1(OC)cc(F)c(CNC2CC2C(=O)Nc2cc(Br)c(C)cc2Br)cc1F 61597,N1(CC(C2CCCOC2)(F)F)CCC(O)C(F)(F)C1 61598,c1(C(N2CC(C(=O)NCCCc3ncc[nH]3)(SC)C2)=O)cc(C)nnc1C 61599,C1(CNC(c2n(C(C)C)ncc2)=O)CN(C(=O)C2=CCCC2)CCC1C 61600,n1(CC(=O)NCC(C2CCC2)NC(C(CC=C)(F)F)=O)cc([N+](=O)[O-])nc1C 61601,Cc1nnccc1C(N1CC2CC1C2NC(=O)C(N1CCCC1)C1CC1)=O 61602,c1(CC)cc(C(=O)NC(C)CC(C)NC(C2CCC(=O)N(C)C2)=O)ccc1O 61603,c1(C(=O)NC2C(CNC(c3cncc(C)c3Cl)=O)CC2)noc2c1CCCC2 61604,N1(C(C2(C3CC3)CNC2)=O)CCCC12CCC2 61605,C1(C(N2CC(C#N)C2)=O)CC(F)(F)CN1C(c1cccc(O)n1)=O 61606,c1(CN(C)C(C2C=CCCC2)=O)cnn2c1CN(C(c1cc(CF)on1)=O)CC2 61607,c1(C(=O)NC2CCCN(C(c3c(C)cccc3O)=O)CC2)ccc2ccsc2c1 61608,CC(C)C(C)CC(=O)NC1CCCC(NC(c2ccoc2C2CC2)=O)C1 61609,c1(OC)cccc(C(N2CCN(C(=O)Cc3cccc(C)c3)C3CC23)=O)c1C 61610,C1(NC(c2ccnc(Br)c2F)=O)COC2(CCC2)C1 61611,c1(OC)ccc2[nH]cc(-c3ccc(Nc4nc(C5CC5)cc(C)n4)nc3)c2c1 61612,c1(N2C(C)C(NC(=O)C(C)(C)F)CC2)nc(Cl)nc2ccc(Cl)nc12 61613,CON=Cc1ccc(C(=O)NCCC(C(C)C)NC(C2CN(C)C(=O)N2)=O)cc1 61614,C#CCC(CC#C)C(=O)N1CCC2(C1)CN(C(C1CC(O)(C#C)C1)=O)C2 61615,N1(C(C2(C)C(CC)CCC2)=O)CCC2(CC1)OC1(CO)CC2(NC(=O)C(C)O)C1 61616,c1(C2(C(N(CC(CNC(Cn3ccc(C)n3)=O)O)C)=O)CC2)ccccc1Cl 61617,C(=O)(C1=NOC(C)C1C)NC(C(C)C)CNC(C1(C)CC1(Cl)Cl)=O 61618,c1(C(N2CC(C(C)NC(Cn3c(C)ccn3)=O)C2)=O)cnnc(Cl)c1 61619,CC1CN(C(C2CCS(=O)(=O)CC2)=O)CCC1NC(=O)CC=CC(C)(C)C 61620,C(C)(C)(CC(=O)NCC1(C)CNC(=O)O1)N(C)C(C1CC2CC2C1)=O 61621,N1(C(C(c2ccccc2)OC)=O)CC(CNC(=O)CC(C)(O)C2CC2)C(C)(C)C1 61622,c1(OCC)ccccc1C(=O)NC(CNC(C1CCCO1)=O)C(C)C 61623,Cc1nnc2c(C(N3CC(C)(NC(c4ccoc4Br)=O)C3)=O)cccn12 61624,C1(CSCC(=O)N(C(CNC(C(=C(C)C2CC2)F)=O)C)C)CCCCO1 61625,CCC(C)CC(=O)NC1CCC1CNC(C1CCN(c2ccc(Cl)nn2)CC1)=O 61626,c1(C(=O)NCC2(NC(COC)=O)CCCC2)cc(Cl)sc1S(N)(=O)=O 61627,C1(CNC(C(=C(C)C2CC2)F)=O)CN(C)CCN1C(c1ccoc1)=O 61628,[N-]=[N+]=NCC(F)CCNC(=O)C(O)CCCNC(c1cnc2n1CCC2)=O 61629,Cc1oc(C(F)(F)F)nc1C(=O)NCC(C(C)C)NC(c1ncn(C)n1)=O 61630,c1(CN2CC(CNC(Cc3cncc(C)c3)=O)C2)c[nH]c2cc(Br)ccc12 61631,O(NC(=O)C(F)C1CCCCC1)CCF.n1(CC=O)[nH]cnc1=N 61632,CC1CN(C(c2ncc(F)cc2F)=O)CCC1NC(c1nn[nH]c1Cl)=O 61633,C1(C(=O)NCC(CC)NC(c2cc(CCO)on2)=O)CCC(O)CN1C 61634,Cc1ccc(NC(N2CCCC(C(C)(C)C)CC2)=O)c(O)n1 61635,N1(C(C2N(C(C(N3CCSCC3)C)=O)CSC2)=O)C2CCC1CC(CO)C2 61636,C1(C(N2CC3(NC(C(CC)C)=O)CC2(COC)C3)=O)CCc2nc[nH]c2C1 61637,Cc1nccnc1C(C(=O)NC1CN(C(=O)OC(C)(C)C)C1)N(C)C1CC1 61638,N1(C(=O)CCc2ccncc2)CCCC2C1CCN2C(c1cnco1)=O 61639,C1(C(N2C(CNC(=O)CC(=O)Nc3nccs3)CC2)=O)CC12CCc1ccccc12 61640,C(=O)(C1=CCCOC1)NCC(C1CCN(C(c2c[nH]cc2C2CC2)=O)CC1)C 61641,CC1CC(NC(C2CCCOCC2)=O)CN1C(C1CC12CCOC2)=O 61642,C1(CC(=O)NC(C(=O)OC)CC2CC2)CCCN(C(=O)C=C(C)C(C)(C)C)C1 61643,c1(C(=O)NC(C)CCCCNC(c2ccc(CO)cn2)=O)n[nH]cc1[N+](=O)[O-] 61644,CC(CC1CCCO1)C(=O)NCCOCCOCCNC(=O)C(c1ccc(Cl)s1)=O 61645,c1(N(CC(=O)NCC(C)NC(=O)C(F)(F)c2nccs2)C)ccccc1 61646,C#Cc1cncc(C(=O)NC2CC(N(C(=O)CCSCc3ccccc3)C)C2)c1 61647,CCC(C)C(CC(=O)NC1CC(C2CC2)C1)NC(=O)COCC(=O)NC 61648,c1(C2CCCN(C(C(=O)NCCCSC)c3ccns3)C2)ccccc1C#N 61649,CC(Cc1ccccc1)C(=O)N(CC(O)CNC(C1CCCC1)=O)C 61650,N1(C(C(C)(C2CC2)NC(C)=O)=O)CCC(CN(C(=O)C(C)CC2CCC2)C)CC1 61651,c1(N(C)Cc2csc(Br)n2)nc(=N)nc(NCCCc2ccccc2)[nH]1 61652,C(CC(C(=O)N1CCCC(OCC)C1)NC(=O)CCCn1ccnc1)OCC 61653,N1(C(C=C(CCC)C)=O)CC2CCCC(CNC(=O)CC3CC(C)=NO3)C2C1 61654,C1(C(=O)NCCCC(C)C)CC(NC(=O)CCC2(C)CC2)CCO1 61655,C1(C(=O)NCC2CC(C(N3C(C)(CC(=O)NC)CC3)=O)C2)CC(N=[N+]=[N-])C1 61656,C1(NC(CC=CC=C)=O)CC(NC(C2CCC(CCCCC)CC2)=O)CC1O 61657,C#CCC(CC(=O)N(C1(c2nn[nH]n2)CCOC1)C1CC1)c1ccccc1 61658,C#CC1CN(C(C2CCC2(F)F)=O)CCN1C(=O)CCOC1CCCC1 61659,n1(CC)cc(CNC(=NCCF)NCc2ccccc2Cl)c(O)nc1=O 61660,Cc1ccc(F)c(C(=O)NCC(C(=O)N2CCC(C(C)C)CC2)C(C)C)c1 61661,N1(C(C2C(CCOC)C2)=O)CCC(F)C(NC(c2cscc2C)=O)C1 61662,C1(CC)(NC(c2ccc(F)s2)=O)CCN(C(=O)CN2CCC2C)CC1 61663,C(=O)(CC(=O)NCCn1cc(CC(C)O)nn1)OC 61664,C1(C)(CNC(CC2N(C(c3scc(C)c3)=O)CC2)=O)NC(=O)NC1=O 61665,Cc1cc(NCCCSCc2ccccc2)ncc1S(=O)(=O)NC1CCC(F)C1 61666,CC1(C)CCC(C)(C(=O)NCCOCCNC(=O)Cc2ccccc2O)CC1 61667,CCCCCC(O)C(=O)NCCN(C(=O)CC1CC(=O)NC1=O)C 61668,C(=O)(CCCC(=O)NCCC1CCCN(C(C2CC3C=CC2C3)=O)C1)N(C)C 61669,c1(C(=O)NC(CN(C(C(COC)(C)O)=O)C)C)coc2c(F)cccc12 61670,c1(C(N2CCCC(F)(CNC(C(C)=C3CC3)=O)C2)=O)cccn2nccc12 61671,N1(C(C(=O)NCc2cccc(OC)c2)c2ccns2)CCSC2COCCC12 61672,c1(CC(=O)NC)ccc(C(=O)NCC2CCN2C(=O)CCn2cncn2)cc1 61673,C12(C(=O)NC(CN(C(C(C)NS(CC)(=O)=O)=O)C)C)CC=CC(C1)OC2 61674,c1(C(=O)NCCN2CCC(NC(C(C)S(N)(=O)=O)=O)CC2)cc2cc[nH]c2cn1 61675,c1(C(=O)NC2CC(CNC(c3ncn(CC)c3)=O)C2)c[nH]c2ccccc2c1=N 61676,N1(C(C2(CCC)CC2)=O)CCC2CCCN(C(c3ccsc3)=O)C2C1 61677,c1(CC)nc(C)cc(=NCC2CN(C(c3nn(CCC)cc3Cl)=O)CC2C)[nH]1 61678,c1(NC(CCN(C(=O)CC(C)SC)CC#C)=O)cccc(F)c1 61679,CC1C(CO)CCCN1CC(=O)Nc1cccc(OC(F)(F)CF)c1 61680,C(=O)(C1=CC(O)C(NC(c2ccc(C)cc2C)=O)C1)NCCOCC(=O)OC 61681,C(=O)(C(F)(F)C(F)F)N1CC2C(CC(=O)NC(c3ccno3)C)C2C1 61682,C1(C(N2CC(C3N(C(C(OC)OC)=O)CCC3)(O)C2)=O)CC(C)CCO1 61683,C(C(O)C(=O)NC1CCC(CCC(=O)NCCN(CCCF)C)C1)=CC 61684,N1(C(C(C)O)=O)CCCC(NC(C2CC3C=CC2C3)=O)CC1 61685,CN1N=C(CC(=O)N2CC3CCN(C(=O)CSC4CC4)C3C2)CC1=O 61686,Cc1cc(CC(=O)NC(C2(O)CN(C(=O)C(F)CC3CCOC3)C2)C)n(C)n1 61687,c1(OC)ccc(CS(CC2(OC(C)C)CCCC2)(=O)=O)cc1Br 61688,c1(OCC)cnc(C(=O)NC2(C)CCC(NC(C3CCCN3C)=O)CC2)c(Cl)c1 61689,Cc1cc(CCC(=O)NCc2occc2C(=O)O)ccc1Br 61690,C1(NC(C2CC(SC)C2)=O)CCCCCCC1NC(=O)CC(C)C(F)F 61691,C1(CCNC(C2(OC(C)C)CCOC2)=O)CN(C(c2cccn2C)=O)CC1C 61692,N1(Cc2ccc(-c3ccc(C(C)(C)C)cc3)o2)C(=O)C2C(O)CCN2C1=O 61693,C1(C(=O)NCC2N(C(C(c3ccc(C)o3)C)=O)CC=C2)CC(S(C)(=O)=O)C1 61694,c1(NCCN(C(C)C)C)cccc(S(=O)(=O)N(C2CC2C)C)n1 61695,C(=O)(C(F)CC(C)(C)NC(=O)CCC(C)(C)N(C)C)N1CCN(C(C#C)C)CC1 61696,c1(C(=O)NCC(N(C(C2CN(C)C(=O)N2)=O)C)C2CC2)c(F)ccc(O)c1F 61697,N1(C(CC(C=C)CC)=O)CC2=C(C1)CN(C(C1CC(OC)C1)=O)C2 61698,C(C)(CC(C(=O)NC1CCCCC1)N(CC(=O)OC1(CO)CCC1)C)SC 61699,N(C(=NCCN(C)C1CC1)NCC(F)F)C1C(OCC)C1 61700,c1(C(C(=O)NCCCSCC)N(CC(C)C)CC)cc(Cl)cc(Cl)c1 61701,C#Cc1cccc(NC(=O)Cc2nc(SC)ns2)c1 61702,CC(C)CC(C(=O)N1CC(NC(=O)CCOCC2CC2)C1)C(C)C 61703,CC(C)C(=O)C(=O)N(C)CC1CCN(C(c2ccnc(C3CC3)c2)=O)C1 61704,N1(C(C(CCCNC(c2c(F)ccc(C)n2)=O)(C)C)=O)CCC2CCC(O)C1C2 61705,C1(NC(COCCOC)=O)CC2(CCCN(C(=O)CC3CCC(F)(F)CO3)C2)C1 61706,CCC(O)C(C)C(=O)NCC1CC(NC(=O)C=Cc2cccs2)C1 61707,c1(CNC(CCn2cc(CC(CC)C(C)C)nn2)=O)nc(OC)ccc1C 61708,C=CCCC(C(=O)NC(C)C(F)F)NC(=O)CCCCNC(N)=O 61709,n1(CCOC)nccc1C(=O)NCC1(F)CN(C(=O)C(O)CC2CCCCC2)C1 61710,C1(C(=O)OCC)CCC(C(=O)NCC2CCN(C(c3sccc3C(C)C)=O)C2)C1 61711,C1(CNC(C2CCS2(=O)=O)=O)CCN(C(=O)C=CCN2CCCC2)C12CC2 61712,c1(C(=O)NC(CN(C)C(C2COC(=O)C2)=O)Cc2ccccc2)ccc(F)cn1 61713,N1(C(C23OCC(C(=O)OC)(C2)C3)=O)CCC2(C1)CN(C(=O)C(C)O)C2 61714,Cn1cnc([N+](=O)[O-])c1NC(=O)C(N1CCC(CCN2CCOCC2)CC1)=O 61715,CC1CC(CO)CN(C(c2ccn(C3CC3(F)F)n2)C(=O)NCC(F)F)C1 61716,C1(C(=O)NC2CN(C(CCC=C)=O)C2)CCCC2(C1)NC(=O)NC2=O 61717,Cc1noc(COCC(N2CC(C(C)NC(c3ncsc3C)=O)C2)=O)n1 61718,c1(C(N2CCCC(C)(CNC(C(C(C)C)F)=O)C2)=O)cc2cc(Cl)c(Cl)cc2[nH]1 61719,N1(C(C2N(C)C(=O)OC2)=O)CCC(F)(C(=O)NCCN2CC3CC3C2)CC1 61720,C1(CCNC(C=C(C)Cl)=O)CN(C(=O)CCCc2ccsc2)CCS1(=O)=O 61721,c1(C(=O)NC(CCNC(C2CC(C)C2)=O)C)cccc(S(C)=O)c1 61722,c1(C(C(=O)NC2(CC(=O)NC(CSC)C)CCC2)F)ccccc1 61723,c1(C(=O)NCC(CNC(=O)CC2CCC3(CCC3)O2)F)cnc(O)c([N+](=O)[O-])c1 61724,c1(C(=O)OCC(c2cc(Cl)cc(Cl)c2)=O)cccc2snnc12 61725,CC1CCCC(C)N(C(=O)CC2CCN(C(C3CCC3C)=O)C2)C1 61726,c1(C(=O)NC(C(C)NC(C2CCCS(=O)(=O)C2)=O)CO)ccc2ncccc2c1 61727,CN1CCN(C)C(C(N2CC(N(C)C(c3ccc(N)c(N)n3)=O)C2)=O)C1 61728,CC(C)C(Cc1ccccc1)C(=O)N1CC(CCNC(C2CCNC2=O)=O)C1 61729,C1(NC(C(C)C(C)O)=O)CN(C(=O)Cc2cccc(O)c2F)CCC12CCC2 61730,Cc1ccc(C(=O)NCC2(CNC(=O)CC3(C)CCCC3)CC2(F)F)c(O)c1 61731,Cc1nn(-c2ccc(Cl)cc2)cc1CN1CCCC2CC12 61732,n1(CC)nccc1-c1cn(CC2CCN2C(C(C)(COC)COC)=O)nn1 61733,CC(=O)C(C)CC(C)C(=O)N1CCCCCC(NC(=O)CC(C)(C)CN(C)C)C1 61734,Cc1nn(C)c(C)c1CC(=O)NCC1CCC(C)CN1C(=O)CCc1cnc[nH]1 61735,CCC(C(=O)NC(CCCNC(=O)Cc1cnns1)c1ccccc1)SC 61736,c1(CC)ncc(C(=O)NC2CCC(CCNC(=O)CC3CC(F)(F)C3)C2)[nH]1 61737,Cc1ccc(C(N2CC(NC(c3cc(C)c(C)s3)=O)C3CC23)=O)cc1C 61738,c1(C(=O)NCCC2CC(OC)CN2C(C2CCNC2=O)=O)c(C)ncn(C)c1=O 61739,C(=O)(CCCC(=O)NCC1(C)CC(NC(c2cc(OC)ccc2N)=O)C1)NC 61740,C(=O)(C1Cc2ccccc21)NCC(CNC(c1cc(C2CC2)ccc1F)=O)O 61741,c1(-c2cn(CCN(C(C(C)Sc3ccc(C)cc3)=O)C)nn2)cc(Cl)ccc1O 61742,C(=O)(CN=c1cc[nH]cc1)N1C(CCNC(C2C(C)SCCC2)=O)CCCC1 61743,C1(NCCCC(c2ccccc2)NC(c2c(C)ccnc2)=O)CCC(C)(C)CO1 61744,C(CC(CNC(=O)Cc1csc(C)n1)NC(=O)CN(C1CCCC1)C)OC 61745,N1(C(C2(C)CCCN(C(=O)CC(F)(F)F)C2)=O)CC2CCNCC2C1 61746,C=CCC(CC)C(=O)NC1(c2ccccc2)CN(C(=O)CC(C)C(F)F)C1 61747,CC1CC(NC(C2CC(n3cnnc3)C2)=O)CCN1C(C1CC(C#N)C1)=O 61748,N1(C(C(C=CCCC)O)=O)CC(C2CCCCN(C(C3(F)CCOC3C)=O)C2)C1 61749,CC#CCCCC(=O)N1CCC(C(=O)NC2(CSC)CC2)C1 61750,C(CN=c1cc(C)nc(N2CCC(NS(C)(=O)=O)C2)[nH]1)(C1CCC1)OC 61751,C1(CNC(C2(OC)CCCC2)=O)CN(C(=O)CCC2CC(C)(C)CO2)CCCO1 61752,N1(C(COC(C)=O)=O)CCCC1C1CCCCN1C(c1cncc(Cl)c1)=O 61753,S(=O)(=O)(c1cccc(F)c1)N(C1CC2CNC1C2)CCCc1cccc(C)n1 61754,C(=O)(CP(C)(C)=O)NCC(C)CN(C(=O)C(C)(C)Oc1ccc(Cl)cc1)C 61755,Cc1noc(N)c1C(=O)NCCN(C1CC1[N+](=O)[O-])C(c1ccccc1)=O 61756,C(=O)(N=c1[nH]nc(CC(C)C)s1)C1(CC#C)CCCCN1C(=O)OC 61757,n1(CCC(=O)NCC2C(NC(c3[nH]c(CC)c(Cl)n3)=O)C2)cnc(C)cc1=O 61758,c1(OC)ccc(F)c(OC)c1C(=O)NCC(C)NC(=O)CCCNC(C)=O 61759,c1(C(=O)NCC(C)(CO)NC(c2ccc(COC)cc2)=O)cncc2c1CCC2 61760,C1(NC(C=CC(CC)C)=O)CCC2CCN(C(=O)Cc3cc(C)cs3)C12 61761,CC1(C)CCN(c2nc(Cl)ncc2C2CC2)CC1CNC(c1ccc(F)cn1)=O 61762,c1(NC2CC(O)(CNC(COc3cc(C)on3)=O)C2)c[n+]([O-])ccc1[N+](=O)[O-] 61763,c1(CC)ncnc(NC(CNC(=O)CN2C(=O)CCC2=O)CC)c1F 61764,C1(F)(CNC(C2C(C)C2(F)F)=O)CCCN(C(=O)CC2(C)CCOCC2)C1 61765,C1(NC(CCOC(C)C)=O)CC2CC1CN(C(c1ncccc1Br)=O)C2 61766,C1(C(=O)NC2CCN(Cc3nc(CC)on3)CC2)CCCN(CP(C)(C)=O)C1 61767,c1(C(N2C(COC)CN(C(C3(C)CCCN3C)=O)CC2)=O)cc(C)c(C)nc1C 61768,C1(O)(c2onc(C)n2)CCN(C2CN(c3[nH]cc(I)c3C)C2)C1 61769,c1(C(N2C(C(N3CC(OC)C(F)C3)=O)C(O)CC2)=O)cnn2ccncc12 61770,C(=O)(C(CCCC(=O)OC(C)(C)C)N1CCC2C(O)C(C)(C)C12)NCCCC 61771,C1(F)(C(N(CC(CC)O)C)=O)CCN(C(=O)C(C)CC(C)C)CC1 61772,S(=O)(=O)(c1nc(N2CCCC2)ccc1Br)N1CC(C)OC(C2CCCC2)C1 61773,CC(C)(CC1CC1)C(=O)NCCNC(C1CC=CCC1)=O 61774,N1(C(C2(C#C)CCCC2)=O)CCN(C)C(C(=O)NC2(CO)CC3CCCC23)C1 61775,c1(C(=O)NC2C(CNC(c3cnc(OCC)s3)=O)C2)ccccc1C(N)=O 61776,c1(OC)noc(C)c1C(=O)N(C)CC1(O)CCN(C(=O)C(c2nc(C)cs2)C)C1 61777,Cc1ccc(N(C(=O)C(C(C)C)NC(=O)Cn2ccccc2=O)C)cn1 61778,C1(C(N2CCC(C(C)(C)CN)CC2)=O)CC(=O)OC1(C)C 61779,c1(C(=O)NCC(CO)NC(C(c2ccccc2)OCC)=O)n[nH]c(C(C)C)n1 61780,C1(COC)CN(C(c2cnn(C)c2C)=O)CCN1C(c1ncccc1Br)=O 61781,c1(OC)cc(CNS(=O)(=O)Cc2ccc(C(F)F)cc2)cc2cc(C)oc12 61782,c1(C(C)C)nc(C(=O)NC2CCCC2C(N2CCCC2)=O)co1 61783,N1(C(CCSCC=C)=O)CCCC(NC(=O)CCNC(=O)NC)C1 61784,C1(CNC(C2(CNC(c3ccc(C)[nH]3)=O)CC(=C)C2)=O)COCC(C)O1 61785,C(=O)(C(C)CC(C)C)N1CC(C(=O)N(C)Cc2cnccn2)(COC)C1 61786,C(C(=O)N1CC(O)(CNC(=O)CC2CC2C)C1)(C(C)(C)C)NC(C)=O 61787,C12(C(=O)NCC34N(C(C5=CC(C)(C)C5)=O)C(CC3)CC4)CCCC1CS(=O)(=O)C2 61788,C(=O)(CCC(C)(C)C(=O)OC)N1C(C)(COC)CC(NC(c2coc(Cl)n2)=O)C1 61789,C(=O)(C(F)(F)C(C12CC3CC1C2C3)OC)NC1CC(CC)(CC)NC1 61790,N1(C(C(N2CCCS2(=O)=O)C)=O)CCCCC1CCCNC(c1ccncc1)=O 61791,c1(CC(=O)NC2CC(NC(=O)CSCc3ccccn3)C2)ccccc1O 61792,CN1CCN(C(=O)C(C(C)(C)C)NC(=O)Cc2cscn2)CC1(C)C 61793,c1(OC)cc(C(N2CC(NC(C3CCOC3C)=O)C(C)(C)C2)=O)cc(N)c1N 61794,Cc1ccncc1-c1ccc(C(N2CCC2C)=O)nc1 61795,c1(SCC(=O)NCCN(C(C2C(C)(COC)C2)=O)CCSC)cc(F)cc(Cl)c1 61796,N1(C(C(N2CC(C)(CO)C2)=O)=O)CCCOCC1 61797,c1(C(C(F)F)NCC(O)COc2ccc(CC(N)=O)cc2)cccc(F)c1F 61798,N1(C(=O)C=C2CCCC2)CCC2(CCCN(C(=O)Cc3ccc(O)nc3)C2)CC1 61799,c1(CNc2cc(OC)c(Br)cc2)cc2c(OCc3ccccc3)c(F)ccc2[nH]1 61800,S(=O)(=O)(c1ccn(C2CC2(F)F)n1)NCC1(C)CNCCC1O 61801,C1(CCC#C)CCCN(C(C2(NC(=O)CCC(C)C)CC(CO)C2)=O)C1 61802,N1(C2CN(C(c3c(C)scc3)=O)C2)CCN(C(=O)COC2CCCCCC2)CC1 61803,n1(CC)nnc(C)c1CNC(C1(CCCO)CCCC1)=O 61804,C12(C(=O)NCC(CN(C)C(C3(CCF)CCC3)=O)O)COCC1C2(F)F 61805,c1(NC(=O)NCC)cccc(C(=O)NC(C2(O)CCN(C(=O)CCOC)C2)C)c1 61806,c1(NC(C(C)C)=O)ccccc1C(=O)NC1CCC(NCc2ncccn2)C1 61807,C1(O)(C(CNC(C2(OC)CC2)=O)C)CCN(C(=O)C(C)(C)c2ccnn2C)C1 61808,N1(C(C2(CC)CCCN2C(C2CCC(C)(C)C2)=O)=O)CC2CC1CN2C 61809,c1(C(=O)NCC2C(C(=O)NCC(COC)C)CCO2)nccc2cc[nH]c12 61810,C(=O)(C(F)C(CC)CC)N(CC(C)O)CCNC(C(C)OCC=C)=O 61811,N1(C(C(C2CCC(=O)N2)C)=O)CCC(C)(NC(c2ncccc2N)=O)CC1 61812,C1(C(=O)NCC2CN(C(CC(C=C)C)=O)C(C)(C)C2)CC2CCC1C21CC1 61813,Cc1ncc(C(N2CCCCC(CNC(C3CC3C3CCCO3)=O)C2)=O)cc1N 61814,C1(CC(=O)NC2CCC(CNC(C3(C=C)CCC3)=O)C2)(C(F)(F)F)CNC(=O)C1 61815,C1(NC(CSCC=CC)=O)CCC12CN(Cc1ccc(NC(=O)C(C)C)cc1)C2 61816,c1(-n2cc(C(CC)(C)O)nn2)cc(C(=O)NC(CO)CC(F)F)ccn1 61817,C1(CNC(C2COCOC2)=O)CCCCN(C(=O)C(F)=CC2CC2)C1 61818,C1(NC(c2c(C)c(O)ccc2)=O)CC2CC(NC(c3ncccc3F)=O)CC2C1 61819,C1(CCNC(C=COCC)=O)CN(C(=O)CCc2scnc2C)CCCO1 61820,c1(OC)cc(Cc2ccnc(O)c2)ccc1C(C)NC(N1CCCC1)=O 61821,N1(C(C(C)(C)O)=O)CCC(c2ccccc2)C(NC(C2(S(C)(=O)=O)CC2)=O)C1 61822,CCC(F)(F)CC(=O)N1CC(CO)(NC(=O)C2=C(Cl)CC2)C1 61823,c1(C(=O)NCC(C2(O)CCN(C(CC3(C=C)CC3)=O)C2)C)cc(OC)cc(Cl)c1 61824,c1(C(=O)NC2C(NC(c3occ(C)c3C)=O)CCC2)cc2c(ncn2C)s1 61825,C1(C(=O)NCC(CNC(C(CCC)(C)C)=O)(C)OC)CCc2cnnn2C1 61826,c1(C(C)NC2CC(c3nnnn3CCCN(C)C)(NC)C2)ccc(-c2cccs2)s1 61827,CC1CN(C(C2CCN(C(c3ccc4[nH]ccc4c3)=O)C2(C)C)=O)CCN(C)C1 61828,C1(N(C)C(C2CCCN2S(C)(=O)=O)=O)CC2CC1N(Cc1ccc(Cl)c(F)c1)C2 61829,CC1(C)CC1(Cl)C(=O)NCCC1CCCN1C(c1cnn(C2CCCCC2)c1)=O 61830,C(C(C)C(=O)NCC(C)N(C(=O)Cc1[nH]cnc1C)C)OCC 61831,c1(C(N2C3C(NC(c4cccc(C)n4)=O)CC(C3)C2)=O)coc2c1C(O)CCC2 61832,S(=O)(=O)(c1c[nH]c(C(N2CCN(C(=O)CN3CC=CC3)C(CO)C2)=O)c1)NC 61833,N1(C(c2nnn(CC)c2C)=O)CCN(C(=O)C=CSC)CC1CF 61834,c1(N(C(=O)NCC2(C(C)C)N=N2)CCO)cccc(Br)n1 61835,n1(CCC(=O)N(C)CCN(C(=O)CCOCC(C)C)C(C)C)ccnn1.CO 61836,C1(CN=[N+]=[N-])CCN(C(c2cn(CCNC(c3c[nH]c(=S)cn3)=O)nn2)=O)CC1 61837,C(C)(CNC(c1cnc(S)nc1)=O)(CC(C)C)NC(CC(=O)NCC)=O 61838,c1(CC)ccc(C(=O)N(C(C)CNC(=O)COc2cc(C)on2)CC)[nH]1 61839,C(=O)(C(C)CCCC(C)C)NC1C(CC)CN(C(c2cc(C(C)C)[nH]n2)=O)CC1 61840,C1(N(C(C2C(CC)CC2)=O)CC)CCC(NC(=O)C(CC2CC2)OC)CC1 61841,c1(C(C(C)C)NC(=O)NC2COCC2F)ccc(C(C)(C)C)cc1 61842,Cc1cc(NC(=O)CCCCCN(C(=O)C(C)S(C)(=O)=O)C)cc(Cl)c1 61843,C1(NC(CC(=C)Br)=O)CC2(C1)CN(C(=O)C=Cc1ccccc1F)C2 61844,CC1CCCn2ncc(C(=O)NC3C4CN(C(C5CC6(C5)CC6(F)F)=O)CC34)c21 61845,c1(C(=O)NCC2CN(C(C(C)Sc3ccc(Cl)cc3)=O)C2)csc2c1CCCC2 61846,C1(C(=O)NC(C)CC#N)CCCCN1C(=O)Nc1ccccc1Cl 61847,c1(CCC(=O)NCCC(N2CCN(C(C3C(=C)C3)=O)CC2)=O)nnc(S)nc1O 61848,C(=O)(C1=NOC(C)(C)C1)NC1N(C(C23CCCC2(C(N)=O)C3)=O)CCC(C)C1 61849,C1(C(N2CCC(NC(C=C(C)C)=O)C(O)C2)=O)CCc2nnc(C)n2C1 61850,C1(CC(=O)Nc2cn(C(C)C)nc2)CCCN(C(C2(O)CCSC2)=O)C1 61851,N1(C(CC(C(C)C)C)=O)C2CCC1C(C)C(NC(C13CC(CC(F)F)(C1)C3)=O)C2 61852,C1(NC(CCOCCOCC)=O)C2CC3CN(C(=O)CC45CCCC4C5)C1C3C2 61853,c1(OC)cc(C(=O)NC(C)C(C)NC(c2cnc(C(C)C)o2)=O)cc(F)c1F 61854,c1(OCC)cc[nH]c(=NCCC(C)NC(=O)C=Cc2cncs2)n1 61855,N1(C(=O)COc2ccc(Cl)cc2Cl)CCC2OCCN(C(C3CC=CC3)=O)C2C1 61856,c1(CNC(CN(S(C)(=O)=O)C)=O)ccc(CNC(C2CCCC2F)=O)cc1 61857,C1(CC(CC)NC(=O)CCc2cnn[nH]2)CCCCC1 61858,c1(OC)cc(N)c(F)cc1C(N1CC2CCC1CN2C(=O)CC1(C)CC1F)=O 61859,c1(CC(N2C(Cn3cc(CCSC)nn3)CCC2)=O)ccc(O)cc1C 61860,C1(COC(C23CCC(C2)C(O)C3O)=O)CC2(CCCC2)CO1 61861,C1(C)(C(N(C(C)(C)CC(=O)NC2C=CCCC2)C)=O)COCCO1 61862,C(C(CC(C)C)C(=O)NCC(C)(O)CC(C)C)NC(c1n[nH]c(CC)c1C)=O 61863,C1(NC(Cc2n(C)ccn2)=O)CC2(CCN(C(=O)C#CC3CCCCO3)CC2)C1 61864,N1(C(c2cc(OCC)ns2)C(=O)NC(C)(C)C)Cc2cccc(F)c2C1 61865,c1(C(=O)NC2CC(NC(c3c(C)c(C#N)ccc3)=O)C2)cncc(P(C)(C)=O)c1 61866,Cc1cnc(C(=O)NCC(C)(O)CNC(c2c[nH]c(=N)s2)=O)cc1Br 61867,Cc1ccc(Br)c(C(N2CC(NC(=O)C3=COCC3)C3CC3C2)=O)c1 61868,C(C(CC1CCCC1)C(=O)N1CCC(C(N)=O)C1)NC(C(OC)OC)=O 61869,c1(CC)ccc(C(N2CC(NC(=O)CC(F)(F)F)C3CC23)=O)cc1[N+](=O)[O-] 61870,CCN=c1cc(-c2nc(Cc3cc(C)c(F)c(F)c3)n(C(C)C)n2)cc[nH]1 61871,C(c1ccccc1C)=CC(N1CCC(CC(=O)N(C2CCN(C)C2)CC)CC1)=O 61872,n1(CC(=O)NCC(C2CCOC2)NC(=O)Cc2cccs2)cc(Cl)cn1 61873,c1(OCCCC(=O)NCCN(C(=O)CC2(C)CC2F)CC)ccc(Cl)cc1C 61874,c1(CNC(c2cc(C)n(C)c2)=O)ccc(CNC(=O)C(F)C(F)(F)F)cc1F 61875,c1(N2CC(C)CN(C)CC2)[nH]c(=NCCS(C)=O)nc2scnc12 61876,C1(CNC(C=C(COC)C)=O)CCCC1C(=O)NC1(C(F)F)CCCC1 61877,C(=O)(CCC(F)(F)C(F)F)NCCCCC(C)NC(CC(C)OC)=O 61878,C(=O)(C1=CC2CCCC12)NCCOCCCN(C)C(c1cnn(C)c1Cl)=O 61879,N1(C(C)=O)CCC(C(=O)N(C)C)CC1.C1(=O)NOCC(=O)NC(C)C12CC2 61880,C1(NC(CCCC)=O)CN(C(C2CCn3c(cnc3C)C2)=O)C2(CCCCC2)C1 61881,c1(C(=O)NC(CC)(C)CNC(=O)Cc2cncs2)cnc(C)c(C#N)c1 61882,C12(C(=O)NCc3c(C(=O)NCC(COC)(C)CO)nco3)CCC(C1)OC2C 61883,c1(C(=O)NCC(C)N(C)C(c2c[nH]c(=O)cn2)=O)cnc(C(F)F)cn1 61884,C1(NC(c2c(CC)csc2)=O)CC=C(C(=O)NCCc2ccon2)C1 61885,n1(CC)cnc2c(N3CCCC4(CC4)C3)[nH]c(=NCC(C(C)(C)C)SC)nc12 61886,C12(NC(C(C=C)CC)=O)CCCC1N(C(C13CC(F)(C1)C3)=O)CCC2 61887,CC12CCN(C1)C(=O)N2.C1CC(=O)N(c2ccccc2F)C1.c1ccccc1F 61888,Cc1cccc(C)c1OCC(=O)NCCC(C)N(C)C(c1cnc(N)c(O)c1)=O 61889,N1(C(c2noc(CC)c2C)=O)CCC2CCN(C(c3c(Br)nnn3C)=O)CC12 61890,CC1(C)CC(NC(c2snnc2C2CC2)=O)CCN(C(=O)Cc2ccsc2)C1 61891,C#CC1CN(C(C2CC2c2ccc(F)c(I)c2)=O)CC1OC 61892,n1(CCC(N2C(C(C)(F)F)CCC2)=O)nc(O)c2c1CCCC2 61893,c1(CNC(C(=O)NC(CCCCC)C)=O)cc(F)ccc1C 61894,c1(NC(C)CC(N)=O)nc2ccccc2nc1N1CC2C(C1)C2(F)F 61895,C1(C(N2C(CC)CC2)=O)CCN(C(=O)Cc2nccn2C)C1(C)C 61896,c1(CNCC(CC2CN(C(CSC)=O)C2)(C)C)cccc2c1oc1ccccc21 61897,Cn1c(O)nc2cc(C(N3C4CCC3CC(CNC(C3CCC3)=O)C4)=O)ccc12 61898,CN(C)S(C)(=O)=Nc1nc(C(=O)NC2(CNC(c3ccncc3O)=O)CC2)cs1 61899,c1(NC(C)CCO)[nH]c(=NCc2nc(Br)n(C)n2)nc2c1cnn2C 61900,N1(C(CCCOCC=C)=O)CCN(C(=O)C(C)c2ccco2)CC1c1cn[nH]c1 61901,C(c1cccnc1)=CC(=O)NCC1CCC(NC(COCc2onc(C)n2)=O)C1 61902,N1(C(C2CC3CCCC3C2)=O)CC2CCCN(C(=O)CSC(F)(F)F)C2C1 61903,C(CS(=O)(=O)CC(=O)N1CCC(C2CC2)C1CNC(c1c[nH]nc1C)=O)OC 61904,C1(NC(C2(N(C)C)CCCOC2)=O)CCCN(c2ccnc(C(F)(F)F)n2)CC1 61905,C1(CNC(C=CCCC)=O)CCCCC1NC(c1cc(CC)c(C)s1)=O 61906,C(=O)(CC1CC(=O)c2ccccc21)NCC1CN(C(CCN(S(C)(=O)=O)C)=O)C1 61907,C(CC(O)CNC(=O)C(C)N(C(=O)CN1CCNC1=O)C1CC1)OC 61908,c1(CN2CCC(C(=O)NCc3ccc(Cl)cc3F)C(O)C2)cc(Cl)c(O)c(Cl)c1 61909,N(C)(C1CCc2c(F)cccc21)C(C(C)C1=CCCC1)=O 61910,C1(C(=O)NCC(CNC(C2C(C(C)(F)F)C2)=O)(C)O)CCCCC(=O)N1 61911,CC1(C)C(NC(=O)CC2CCCCC2)CCN1C(=O)CC(F)(F)Cl 61912,N1(C(C)=O)CC(NS(=O)(=O)CC)C(C)(C)C1.C(=O)(CCO)NCC(C1CCCC1)OC 61913,C1(CNC(c2c(OC)c(Br)sc2)=O)(CO)COCC2CCCCN12 61914,c1(C(=O)NCC(c2ccco2)OC)n[nH]c2c1CN(C(=O)C(C)CC1CC1)C2 61915,C1(C(=O)NC2(CC)CC2)COC2(C1)CN(C(C1OCCC1(C)C)=O)C2 61916,c1(C(N2CC(C)C(CNC(C3CCC=CO3)=O)C2)=O)cccc(Cl)c1N 61917,c1(NC)ccc(C(N2CCN(C(C3Cc4nnsc4S3)=O)CC2C)=O)cc1F 61918,CC(CN=c1nc(C2CCCC2)[nH]s1)NC(N)=O 61919,C1(CNC(C2CCCC3CC23)=O)CCN(C(c2nnc(O)nc2O)=O)C12CC2 61920,c1(C(N2CCN(C(CCC=CC(C)C)=O)C(C)C2)=O)cnc2c(C#N)cnn2c1 61921,c1(C(N(C2CCCC2)CC#CC)=O)ccc(NC(=O)CC(C)n2ccnc2)s1 61922,c1(C(=O)NC2CC(C)N(C(=O)C(C)n3cccn3)C2)nc(F)ccc1Cl 61923,C1(C(=O)NCCC(=C)CNC(=O)C=Cc2cnc[nH]2)CCCC(=O)N1 61924,c1(-n2c(CC3CC(C)C3)nc(CC(C)(C)CO)n2)nc2ccccc2n(C)c1=O 61925,C(=O)(C(C)(C)CN=c1[nH]c(=NCCS(=O)(=O)CCO)c2cccc(F)c2[nH]1)NC 61926,C1(NC(=O)COCc2ccncc2)C2CN(CC(=O)NCCC3CCOC3)CC12 61927,C1(C(=O)NCCC2CCC(C(F)F)CC2)CC(C2CCC2)C1 61928,Cc1c(CC(=O)NCC2CC2NC(=O)C2=CC(C)(C)C2)c(O)nc2[nH]nc(O)c12 61929,CON(C)S(=O)(=O)c1cccc(C(N2CC3CC2C3NC(C2CC(F)C2)=O)=O)c1 61930,Cc1cc(C(=O)NCc2cccc(C(=O)NC(C)C(F)(F)Cl)n2)c(C)s1 61931,CC1(C)CCN(C(C2CSCCS2)=O)CC1NC(c1coc(Cl)n1)=O 61932,CC(C)(O)C(c1ccccc1)C(=O)NC(=O)CN1CC(n2cccn2)C1 61933,C(N=c1ccc(C#N)c[nH]1)C1OCC(CNC(c2c(Cl)cn(CC)n2)=O)C1 61934,Fc1ccc2c(c1)C(N=c1ccnc(NCCC3CCCO3)[nH]1)CCO2 61935,Cc1ccc(-c2cn(C(C)CC3(CNC(=O)C(C)N(C)C)CC3)nn2)c(F)c1 61936,c1(CC(=O)NCC(CCNC(CCC=CC)=O)(C)C)coc2c(F)c(F)ccc12 61937,C(C(C)C(F)(F)F)NC(CCC1CCC(NC(C2(C=C)CCC2)=O)C1)=O 61938,c1(C(=O)NC(C2CN(C(=O)CC3CCOC3=O)C2)C)cnsc1C 61939,CCN=C(NCCS(=O)(=O)c1ccccc1C)N1CCC2(CCCC2)C1 61940,CCC(C)C(C(=O)NC1CN(C(=O)Cc2ccnc(OC)c2)CC1C)N(C)C 61941,CN1CCN(C(C2CNC(=O)N2)=O)CC1CNC(c1ccc(-c2ccco2)o1)=O 61942,Cc1oc(S(N)(=O)=O)cc1C(N1CCN(C(C2CCC3(CCC3)C2)=O)C(C)C1)=O 61943,CCS(=O)(=O)c1cnc(O)c(C(=O)NCCC(C)CCNC(C2(C#N)CC2)=O)c1 61944,C(=O)(C(C(C)(C)C)NC(C1CNC(=O)C1)=O)NC(CCSC)C 61945,C#CC1(NC(=O)CC2(CNC(=O)C(C)=CC(C)(C)C)CC2)CCC(C)(C)C1 61946,c1(C(=O)NC2CC3CC(NC(C(C(=C)Cl)(C)C)=O)CC32)cc(F)c(F)c(C#N)c1 61947,c1(C(=O)NC2(CO)CN(C(CC3CNC(=O)O3)=O)C2)cc2n(n1)CCO2 61948,S(=O)(=O)(CC(C)(C)C(C)C)NCC(n1cc(CCCC=C)nn1)C 61949,c1(C(C)C(=O)N(CCCC2CCCN2c2cc(F)ncn2)CCO)ccc(F)c(F)c1 61950,c1(OC)cccc(C2(C(=O)NCCN(C)C(C3CC=CCC3C)=O)CC2)n1 61951,c1(CN(C2CCC2)C)ncc(-n2cc(-c3ccc(C(=O)O)cn3)nn2)cn1 61952,C1(C(=O)NC2(C)CN(C(C(C)SC(F)(F)F)=O)C2)CCN(C(=O)C(N)=O)CC1 61953,c1(C(=O)NCC(CNC(c2c(COC)cco2)=O)F)ccc2c(c1)COC2 61954,CCC(CC(=O)NC1CCC(O)CN(C(=O)Cc2cccc(OC)c2)C1)C(C)C 61955,c1(C(=O)NCCC23C(CN(C(C(C)(C)C(F)F)=O)C2)CC3)cnc2occc2c1 61956,C1(C(C)C(=O)NCC(C2CC2)NC(C2CCC2CF)=O)CCCCC1 61957,CCCCC(C(=O)N(C)CCC1CCCCN1C(=O)CN(C1CC1)CC)C(C)C 61958,c1(C(=O)NCC(C)NC(=O)C(C)CC2CCCCC2)nc(Br)n2ccccc12 61959,N1(C(CCN(CC)CC)=O)CC2CCC2(CNC(c2c(C)ccn2C)=O)C1 61960,C1(C(=O)NCC)(C(C)C)CCCN(C(c2cccc(OCC)c2O)=O)C1 61961,C1(NC(=O)NCC(c2ccccc2)C)CCCCC1N=c1ccnc(CO)[nH]1 61962,n1(CCC(=O)NC(CC=C)CNC(=O)C(F)(F)C(C)O)nc(O)c2ccccc12 61963,N1(C(c2ccnc(C(=O)OC)c2)C(=O)NCCOC)CCCC(O)(C(C)C)C1 61964,N#Cc1cc(C(N2CC(NC(C3CCCOC3)=O)CC(F)C2)=O)ccc1F 61965,n1(CC(=O)NCC2CN(C(=O)C(O)CC3CCOCC3)CCO2)ncccc1=O 61966,CC1(C)CCOC1C(=O)NCC1(C(=O)Nc2cncc(Cl)c2)CC1 61967,C(CCCC(CO)NC(=O)C(O)Cc1cc(Cl)sc1Cl)NC(=O)COC1CC1 61968,C(=O)(C(C)(F)C(=O)Nc1cccc(NC(C2(C)C=CCCC2)=O)c1)OCC 61969,c1(CC(N2CC(COC)(CNC(=O)CC3CCCC3(F)F)C2)=O)ccc(F)cc1Cl 61970,N1(C(=O)Nc2cccc(OCC)c2)CC(=O)Nc2ccc(C#N)cc21 61971,c1(C(=O)NC(C(C)C)CNC(=O)CCc2cncnc2)cccnc1O 61972,C(=O)(C(O)C1=CCCCC1)NC(C(=O)NCC(C#C)OC)CC(=C)Cl 61973,c1(CCC)ncoc1C(=O)N(C)CCNC(c1cnn(C(F)(F)F)c1)=O 61974,CC(CC(C)NC(=O)Cc1cnn2ccccc12)N=c1[nH]c(Cl)nc2c1SCC2 61975,CC(C)C(C)CC(=O)NC1(C2CCCN2C(=O)CN2C(=O)CCCC2=O)CC1 61976,c1(NCC2CCCN(C)C2)ccc(S(=O)(=O)NCCOC2CC2(F)F)c(Cl)c1 61977,C1(C)(CCOC)CN(N2CCCC(c3nc(C)c(C)[nH]3)C2)C1 61978,C(C(C)(C)CNC(=O)CN1CCCC1CO)N(C(CN(C1CC1)CC)=O)C 61979,C1(NC(c2nc(C3N(C(C)=O)CCC3)sc2)=O)CCC(NC(C2(C)CC2)=O)CC1 61980,c1(C(N2CCC(NC(=O)C=Cc3ccccc3)CC2)=O)cc(NC2CC2)ncc1Cl 61981,C12(NC(c3c(CC)csc3)=O)CCCC1CN(C(=O)C(C1CC1)C1CC1)C2 61982,N1(C(C(C(CC)C)N)=O)CCC2CN(C(=O)Cc3cccc([N+](=O)[O-])c3)CC12 61983,C1(CCC)CN(C(c2cc(OC)ns2)=O)CC1C(=O)NCC1CC(=O)N(C)C1 61984,C=C(Br)CN=C(NCC(=O)NC1CCCCO1)NCC(=O)NCC(F)F 61985,N1(Cc2nc(C)sc2)CCCC(O)(CNC(=O)C(=O)C(C)C)C1 61986,c1(OC)ccc(CN(C(c2ccccc2OC)C(=O)NC2CCCC2)C)nn1 61987,CCC(C(=O)OC)C(=O)NC1CC1NC(c1cn(C(C)(C)C)nn1)=O 61988,c1(C2CN(C(C=CC(C)(C)SC)=O)C2)cc(O)n[nH]1.C1(N2C(C)C2=O)CC(C#N)C1 61989,O(NC(=O)CCCN(C)C(C1CC(C)(C)CN1C)=O)CC(=C)C 61990,N1(C(c2c(N)ccc(C)c2)=O)CCC2(CCN(C(C3(C(N)=O)CC3)=O)C2)C1 61991,C1(C2(NC(C3(C(=O)OC)C=CCC3)=O)CC2)CCCCN1C(c1ncncc1Cl)=O 61992,CC1(CNC(C23CCCC2CCC3)=O)CCCN(C(c2cc(N)c(F)cn2)=O)C1 61993,c1(CC(=O)Nc2occ(COC)n2)c(C)nc(-c2ncccn2)nc1O 61994,C1(C)(NC(C2CC(=C)C2)=O)CCN(C(=O)CCn2c(-c3cccs3)nnc2S)CC1 61995,n1(C(COC)C)nc(-c2ccoc2)nc1Cc1noc(CCC(C)C)n1 61996,CC(C)CC(C(=O)N1CCC(CCN(C)C(C2(C)C=CCCC2)=O)CC1)N(C)C 61997,CC1N(C(c2ccc(CNC(c3cc(C#N)cs3)=O)o2)=O)CCCC1(C)C 61998,C=C(C)C(CC(=O)N1CCC(NC(=O)CN2CCC(CC)C2C)CC1C)OCC 61999,c1(C(N2CCC(CCN(C)C(C3(C4CC4)CC3)=O)CC2)=O)cccc2sccc12 62000,C1(C)(OCC(=O)N(C(C#C)C)CC)CN(C(=O)Cc2sccc2C)C1 62001,N1(C(=O)Cc2cc[nH]c2)CC(C2CCCN(C(=O)C(O)C3CCC3)C2)C1 62002,Cc1cc2n(n1)CCCN(C(c1nccc3occc13)=O)C2 62003,C(C(CNC(C1C2(CC2)C12CC2)=O)S(C)(=O)=O)NC(C(c1c(C)cccc1)C)=O 62004,c1(CN2C(C(=O)Nc3c(C(C)C)scn3)CC3CC32)ccc(O)c(Cl)c1 62005,N1(C(c2cc3cccnc3s2)C(=O)NCCCC)CCNC(=O)C(F)(F)C1 62006,C1(CC)(CC)CC(NC(=O)Cc2nonc2C)CN1C(c1ccc(C)s1)=O 62007,c1(C(N(CC(O)CN(C(=O)C=Cc2cn[nH]c2)C)C)=O)cccc(F)c1[N+](=O)[O-] 62008,C1(C(=O)NCC2CCC(N(C)C(C3CC3C3CCC3)=O)CC2)Cc2nncn2C1 62009,N1(C(c2occ(C)c2)=O)CC=C(CC(=O)N(C2CCN(C(C)C)C2)C)CC1 62010,c1(C(=O)NC2CCC(CS(C)(=O)=O)CC2)cc2cc3c(cc2[nH]1)OCCO3 62011,C1(O)(C(C)NC(C(CSC)C)=O)CCN(C(c2cc(Cl)cnc2C)=O)CC1 62012,C1(C(N2CCC(C(=O)OC)CC2)=O)CN(C(c2ccno2)=O)Cc2cccn2C1 62013,O=C(C(F)(F)C(F)c1ccccc1)NC(c1ccc(F)cc1)c1ccc(Cl)cc1 62014,c1(C(C)N(C(N)=O)CC2CCCCO2)ccc(CNC(=O)CCc2cnc[nH]2)cc1 62015,CC(O)C(F)(F)C(=O)N1CC=CC(C(=O)NCc2cncnc2)C1 62016,c1(CC(=O)NCC2CCC2NC(C2CC3CC3C2)=O)c[nH]c2cccc(F)c12 62017,c1(N2CCC(C=C)C2)nc(N2CCC3(CCC(O)C3)C2)nc2ccsc12 62018,c1(C(=O)NCCn2cc(CNC(COCCC)=O)nn2)cc(F)ncc1OC 62019,C1(NC(c2cnc(Cc3ccc(OC)cc3Cl)s2)=O)(CO)CCCC(C)(C)C1 62020,c1(N2C(CNCc3ccc(C(=O)OCC)o3)CCC2)ncnn2cc(Br)cc12 62021,c1(CC)c[nH]c(C(=O)NCC2C(CNC(=O)CC(=O)N(C)C)C2(F)F)c1 62022,c1(C(=O)NC2CCCN(c3nc(O)n[nH]3)C2)c(Cl)cc(F)cc1Br 62023,Cc1nsc(N(C)CCOCCNC(C2CCC(C)O2)=O)c1C#N 62024,N1(C(=O)Cc2cn[nH]c2)CCC(OCCNC(=O)CCCC2CCCO2)C1 62025,c1(SCC)ccc(C(N2CCC(F)(C(=O)N(C)C)C2)=O)cc1 62026,CC1CC(=O)NCC1C(N1CCCN(C(=O)CCN2CCC(O)CC2)CC1)=O 62027,C1(C(=O)NCC(=C)C)CCN(C(C2CCN(C)C(=O)C2)=O)CCO1 62028,N1(C(c2ccccn2)=O)CC2(C1)CN(C(=O)CNC1C(C(C)(C)O)C1)CC2CO 62029,N1(C(Cc2cn(CC)nc2)=O)CCCC(C(N2CCC(OC)CC2)=O)C1 62030,N1(C(C(C)SC)=O)CCCC(C)(C)C1C(=O)NCC1CCCN1C 62031,CN1C(=O)OC2CN(C(C3CCCC(NC(=O)C(F)F)CC3)=O)CC12 62032,c1(C(=O)NCCC2N(C(C(=O)NC3CC3)=O)CC(F)(F)C2)c(F)ccc(F)c1Cl 62033,CCCCCCC(=O)NC(C1CCCC1)CNC(c1ccncc1C(F)F)=O 62034,Cc1cc(C(N2CCC(NC(C3CC4(C3)CC(F)(F)C4)=O)C2)=O)c(N)cc1F 62035,CC1CN(C(=O)Cc2ccsc2)CC(CCNC(c2cnc(C(C)(C)C)o2)=O)O1 62036,C(=O)(C1=CCCC1)NC(CC)CN(C(=O)C(c1ccccc1)OC)C 62037,c1(C(=O)NCC2C(NC(C(C(C)C)(C)O)=O)CCC2)cccc2cc[nH]c12 62038,C1(C(N2C(C3(NC(Cc4n(C)cnc4)=O)CC3)CCC2)=O)OCCOC12CCC2 62039,C1(CC(N2CCN(C(c3c[nH]c(=N)o3)=O)CC2)=O)Oc2ccccc2NC1=O 62040,N1(CC2(C(=O)O)CC(=C)C2)CC2(C)CC1CCO2 62041,c1(OC)cc(C(=O)NCC(C(C)C)NC(C23CCC(F)(CO2)C3)=O)cnc1OC 62042,c1(CC)c(C(N2CCCCC2Cc2cn(Cc3ncc(Br)n3C)nn2)=O)csc1C 62043,c1(CC(C)NC(c2c(F)cccc2F)CCOC)ccc(OC)c(F)c1 62044,C1(C)(C(C)C)CCN(C(CCc2cnn(C)c2)C(=O)NCCCOCC2CC2)C1 62045,N1(C(C2CCC(Nc3ncnc4ccccc34)CC2)=O)CCC2(CCCOC2)C1 62046,CN1CCN(C(C(=O)N(CC)CC2CCCO2)c2ccco2)C(c2ncc[nH]2)C1 62047,C(=O)(CCCCC(C)(C)C)N(C1C2CCCC12)C 62048,C1(C)(C(=O)NCC(=C2CN(C(CC(C)C3CC3)=O)C2)F)CCOC(C)C1 62049,Cn1cnc2[nH]c(C(=O)NC3(CNC(=O)C(C)(C)F)CCC3)cc12 62050,c1(C(=O)NC(C(C)NC(c2ccn(CCF)n2)=O)C)cccc2cncn12 62051,N1(C(=O)CCN2C(=O)CCC2=O)CCC2CCN(C(c3cncc(Cl)c3)=O)C2C1 62052,C(=O)(C#CC1(C)CC1)N1CCC(C)(CCNC(C2CN(C)C2)=O)C1 62053,c1(CCC(=O)NCC2CC2NC(=O)CC2CNC(=O)C2)cccnc1Br 62054,CCCCCCCCC(=O)NCCOC(c1cccc(S(=O)(=O)N(C)C)c1)=O 62055,C(=O)(CC(C(F)(F)F)NC(=O)Cc1cccnc1O)NCCSCC#C 62056,C#CCC(C)(C(=O)NCCCC(C)CO)NC(=O)Cc1cccn1C 62057,C1(C(=O)NC2C(NC(c3cc(O)ncn3)=O)CC2)CC(c2cccnc2)=NO1 62058,c1(-c2nc(CNC(C(=O)NCC(CC)(C)CC)=O)sc2C)ccc(C)c(F)c1F 62059,Cc1cccc2c(C(=O)NCC3(C)CCCN(C(c4ccnnc4)=O)C3)coc12 62060,C(C(C)(O)C(=O)N1CC(CC(F)C(=O)OC)C1)C(=O)NC 62061,C1(NC(CCC=C(C)C)=O)CC(C(=O)NC2CCC(O)C(O)C2)C12CCC2 62062,N1(C(CC(COC)NC(=O)CCc2ccc[nH]2)=O)CC2(CNC(=O)OC2)C1 62063,C1(CC)CCc2sc(C(=O)NCC3(O)CN(C(C4CSCCS4)=O)C3)cc2C1 62064,n1(C(C=C)C)nc(-c2ccsc2)nc1-c1nn(C)nc1Br 62065,C1(CCN(C)C)CC(C(=O)N(C)CCNC(=O)CNC(=O)OC(C)(C)C)C1 62066,C(c1ncc[nH]1)=CC(=O)NCC(CO)NC(=O)C=CC1CCOC1 62067,CC1CNC(=O)CN1C(C1CC(CNC(C2CC(F)(CF)C2)=O)C1)=O 62068,Cc1cc(C)c2[nH]cc(C(N3CCC(O)(C(F)(F)F)CC3)=O)c(=O)c2c1 62069,N1(c2nccc(-n3c(C)cc(C)n3)n2)CCC(NC(c2cccnc2)=O)C(O)C1 62070,C(CCC(CCC)NC(=O)CC1CC(OC)C1)NC(C(F)=CC)=O 62071,CC1(C)COC(CC(=O)NC2CC(NC(=O)C=C3CCC3)C2)CO1 62072,C(=O)(C1=C(C#N)CCC1)N1C(CNC(COc2cccc(C)c2F)=O)COCC1 62073,CCC(C)(C)C(O)C(=O)N1CCC2CC1CN2C(c1cccc(F)c1Cl)=O 62074,N1(C(c2c(OCC=C)cccn2)=O)CCC2(CC1)CN(C(C1CCC3CC13)=O)C2 62075,C1(CN(C)C(C2(CN(C)C)CC2)=O)COCCN1C(=O)CCc1cncc(F)c1 62076,C1(C(N2CCC(O)(CO)C2)=O)(CNC(=O)C(O)CC2CCCC2)CC(F)(F)C1 62077,CC1(C)CC(NC(c2[nH]ccc2Cl)=O)CC(C)(C)S1 62078,c1(CC)ncc(C(=O)NC(C)CCN(C(=O)Cc2cccc(O)c2F)C)c(C)n1 62079,N1(C(c2cccc(I)c2)C(=O)NCC(=C)C)CCN(C2CCCC2C(N)=O)CC1 62080,CCCCC(C(=O)N1CCN(C)CC1C(=O)NC(CCC)c1nn[nH]n1)C(C)C 62081,c1(C(=O)OC)ccc(O)nc1N1CCC(CCNC(=O)C(=O)NCC2CC2)C1 62082,C1(CCNC(CC(=O)OC)=O)CN(C(c2cc(O)n(C)n2)=O)CCCO1 62083,N1(C(c2ccc(CSCCC)o2)=O)CCC(CNC(C2SC3C=CC2C3)=O)CC1 62084,C1(NC(COC(CC)(C)C)=O)CN(C(=O)C=Cc2ccccc2C)C2CCCC12 62085,N1(C(C=COCC)=O)CCC2(CC1)CCN2C(c1cccc2[nH]ncc12)=O 62086,C1(C(=O)NCC(C2CCN(C(C(C)n3cccn3)=O)CC2)O)CC(=O)NC(=O)N1 62087,c1(C(=O)NC(C2CCN(C(=O)CN(C)C(c3cccs3)=O)C2)C)ncc(Cl)s1 62088,c1(C(=O)Nc2nc(C(=O)NCCC#C)n(C)c2)c(C)cc(OC)cc1C 62089,C(CC(CNC(c1cnnn1-c1ccccc1)=O)NC(=O)CC1(C)CCC1)OC 62090,Cc1cnc2nccc(C(=O)NC(CNC(C3(O)CCSC3)=O)C(C)(C)C)c2c1 62091,Cc1nn(C(C)C)cc1C(=O)N(C1CC(NC(=O)C(C)(O)C2CCOCC2)C1)C 62092,O=C1NCc2ccc(C(N3CC(NC(c4csc(C(F)(F)F)c4)=O)C3)=O)cc2N1 62093,CC(C(=O)NCC1(C(N)=O)CN(C(=O)CC2CCCC(F)(F)C2)C1)S(C)(=O)=O 62094,Cc1csc2cc(CNC(=O)NC3CC4CC3CN(C(=O)OC(C)(C)C)C4)[nH]c12 62095,c1(OC)cccc(OC(F)F)c1CNC(=NCCOC)NCCC1CCCO1 62096,Cc1cc(C)c(OC(=O)C(O)CC[S+](C)C)c(Br)c1C 62097,Cc1ccccc1CC(=O)N(C1(C(N2CCC2CO)=O)CC1)C 62098,C1(CC=C)(NC(c2cccc(CF)c2)=O)CCN(C(C2OCCO2)=O)C1 62099,Cc1cccc(C)c1CCN=C(NCc1ncccc1Cl)NC1CCN(C(C)=O)C1 62100,c1(C(=O)NC23CC(NC(c4csc(C(F)F)c4)=O)(C2)C3)cc(Cl)c2n[nH]cc2c1 62101,c1(N(C)C)ccc(-c2nc(CCc3nccn3C)n(CC(C)(C)C)n2)cn1 62102,c1(C(=O)OCC)nc(=NC(C)CNC(=O)Cc2cccnc2)cc(C(C)(C)C)[nH]1 62103,c1(OC)cc(C(=O)NCCC(C)NC(C2CNC(=O)C2)=O)cc2c(C)c(C)[nH]c12 62104,N1(C(C(F)(F)C2(OC)CCC2)=O)CC(N(C)C(C2CC3(CC3)CO2)=O)C(F)C1 62105,c1(C(=O)OC)ccc(C(=O)NC2CC2NC(C23CCCC2C3(F)F)=O)c(C#N)c1 62106,CC1CN(C(=O)COc2ccon2)CC(C)N(C(c2cc3cccnc3[nH]2)=O)C1 62107,c1(C(=O)NC2C(C)CN(C(C3CC=CCC3)=O)C2)cn2c(n1)SCC2 62108,C#CCCCC(C)C(=O)NCC(CC=C)C(=O)N1CCC(CN=[N+]=[N-])C1 62109,C12(CNC(C3N(C)CCC3)=O)CC1CN(C(=O)CCNC(=O)C=CCl)C2 62110,N#Cc1cccc(NC(=O)CC2(NS(=O)(=O)c3cn[nH]c3)CCC2)c1[N+](=O)[O-] 62111,N1(C(C(c2ccc(F)cc2)OC)=O)CCCCC1C(=O)OCC(C)N(C)OC 62112,Cn1cc(C(N2CCC(C(F)CNC(=O)CCS(C)=O)CC2)=O)c(Cl)n1 62113,c1(C(N2CC3(CN(C(c4c(C)ccnn4)=O)C3)C2)=O)cccc2cnccc12 62114,C(=O)(CCCCCC#N)NC(C(C)O)C(=O)NC(CCO)C(C)(C)C 62115,CC(C)(C)C(CC(=O)NCc1cccc(NC(=O)CC=CC(C)(C)C)c1)C(F)F 62116,Cc1ncc(Cl)c(C(=O)NC2CC23CCN(C(c2ccncn2)=O)C3)n1 62117,C1(CC(N2CC(CNC(C(CCC)OC)=O)(OC)C2)=O)CCCCC1(F)F 62118,Cc1cc(C(N2CCN(C(C3(c4ccc(O)cc4)CC3)=O)CC2C)=O)cnc1Cl 62119,Cc1cc(C)c(C(=O)NC(CNC(C2(C)CC2C(F)(F)F)=O)C2CC2)[nH]1 62120,C1(C(N2C(CC(N3CC(C(N)=O)(OC)C3)=O)CC2)=O)C2CC3C(C2)C13 62121,c1(CC(=O)NC2CN(C(c3c(=N)[nH]cnc3)=O)C3C2C3)ccc(F)c(Cl)c1 62122,C(=O)(C(C)S(C)(=O)=O)N(CC(C)CNC(=O)COc1nn(C)cc1Br)C 62123,C(=O)(CCCC(=O)NC(C1COCCO1)C1CC1)NC 62124,c1(C(=O)NC(C)(C)CCNC(=O)C2=CCC2)cc(C(F)F)cc(C(F)(F)F)c1 62125,c1(C(=O)NC(C(C)C)CNC(c2cccc(Cl)c2Cl)=O)nccc(C#N)c1F 62126,N1(C(COCCC=C)=O)CCC2CCN(C(=O)C(c3ncccc3C)(F)F)CC12 62127,CC(C)C(C(=O)NC1CCN(C(=O)C=Cc2cccc(CO)c2)C1C)C(C)C 62128,CCCCC(CNC(c1cnc(O)o1)=O)NC(C1(CC)CC1(F)F)=O 62129,C1(NC(C(C=C)O)=O)C2CC1N(C(C1(S(C)(=O)=O)CC1)=O)C2 62130,c1(C(=O)CC(F)F)cc(C(=O)NCC2CCCN(CC(F)(F)F)C2)cc(F)c1 62131,N1(C(c2ccn(C3CCCC3)n2)=O)CCOC(CCN(C(C2(O)CC2)=O)C2CC2)C1 62132,c1(CSCC(=O)OCC2CCOCO2)ccc(N2N=CCC2=O)cc1 62133,c1(C(N(C(CCNC(c2c(C)[nH]nc2Cl)=O)C)C)=O)ccc(S(C)=O)cc1 62134,C1(CNC(c2nn(C)c(Br)c2)=O)CC2(CCC2)CN1C(=O)C(F)=C1CCC1 62135,C1(CC#C)(C(=O)NCCC(C)CCNC(c2c[nH]cc2C)=O)CCOCC1 62136,c1(CNC(C2(NC(=O)CNC(N3CCOCC3)=O)CC2)=O)cncc(Cl)c1 62137,C(=O)(C(C)(O)C(F)(F)F)N(C1CCCN(C(C23CC(CN2C2CC2)C3)=O)CC1)C 62138,Cc1cc(C)c(C(=O)NCC2(O)CN(C(=O)CC(C)c3ccccc3)C2)cc1N 62139,N1(C(CC(C)OC)=O)CCC(NC(=O)CSc2nnnn2C2CCCC2)C12CC2 62140,Cc1ccc(N)c(C(N2CC(O)(CCNC(C3CC(C)CC(=O)N3)=O)C2)=O)c1 62141,CCCC(C)(CCC)C(=O)NCCOC1CCN(C(C2CCCCS2)=O)C1 62142,C#Cc1cc(C(=O)NC2CCN(C(c3cnc(N(C)C)cn3)=O)C2)cc(F)c1 62143,C#CC12CC(CN1C(C1CCOCC1NC(=O)C(C)CC(C)C)=O)C2 62144,C(C(=O)N=c1cc(C(N)=O)n(C)[nH]1)C1N(C(C(CCC)(F)F)=O)CCC1 62145,C1(C(=O)NCC(C)N(C(=O)C=C2CCN(C)C2)CC)CCOC2(CCC2)C1 62146,c1(CNC(=O)CC2CCN(S(=O)(=O)CCCN3CCOCC3)C2)ccnc(F)c1 62147,c1(OC)cc(C=CC(N2CC(C)CCC2Cc2ccccc2)=O)ccc1F 62148,c1(C(N2C(C(=O)NC(CC)CC)CC(C)C2)=O)cc(OC)cc(C(F)(F)F)c1 62149,c1(OC)cc(C(=O)NC(C)Cc2ccc3c(c2)CCC3)nc2ccccc12 62150,C1(c2n(CC(=C)C)nnn2)(NCCCCO)CC2CCC(C1)N2CCC 62151,C1(NC(c2c(CNC(Cn3c(C)ncc3)=O)c[nH]n2)=O)CCSC(C)C1 62152,C1(NC(C2CN(C)C2)=O)CCN(C(c2cn(C)c(=O)cn2)=O)CC1O 62153,C1(C(=O)NCC(CC(C)C)NC(=O)C(C)n2cccn2)CC(S(C)(=O)=O)C1 62154,C1(F)(CNC(C(CC)c2ccccc2)=O)CCN(C(c2sccc2C)=O)C1 62155,N1(CCNC(c2c(CC)nccn2)=O)CCCN(C(c2cccs2)=O)CC1 62156,c1(CC(=O)OCC)ccc(NC(CNC(=O)COCCCC(C)C)CC)cc1 62157,C#CC1CCCN(C(c2ccc(C(=O)OCC)cn2)C(=O)NCCC#N)C1 62158,c1(CC(N2CC(C)C(NC(=O)CN(C)S(=O)(=O)N(C)C)C2)=O)cc(F)ccc1O 62159,N1(C(C2C(C=C)OCC2)=O)CC(CNC(=O)CCc2cnc[nH]2)CC1(C)C 62160,c1(CNC(c2ccccc2F)(C(=O)OC)C)cc(Cl)c2c(c1)OCCO2 62161,c1(C(C)=O)ccc(C(=O)NCCCC(C)NC(c2cc(-c3ccco3)no2)=O)o1 62162,N1(C(c2ccn(CC)n2)=O)CC(CNC(c2c(C3CCC3)cnn2C)=O)C(C)C1 62163,c1(C(N(CCC(F)(F)F)C(=O)C2CC2)=O)cccnc1SCC(=O)NCC 62164,C1(OC)CCCCN(CC(N2CC=CC23CCCC3)=O)C1=O.C(CO)N 62165,C(N=c1[nH]cnc(Cl)c1C)c1ccc(CNC(c2c(N)ncc(C)c2)=O)c(F)c1 62166,c1(C(=O)NCC2(O)CN(C(c3c(SC)n(C)nc3)=O)C2)ccnn(C)c1=O 62167,CCCC(CNC(c1cn(C2CCOC2)cn1)=O)NC(C12CSCC1C2)=O 62168,c1(N(S(CCC(=O)OC)(=O)=O)C2CCNCC2(C)C)ncc(C#N)c(OC)n1 62169,Cc1cc(S(=O)(=O)N2CC(N3CCCNC3=O)C2)ccc1OC(F)F 62170,N1(C(c2cccc(-c3ccccc3)n2)=O)CC2CC1CN2C(C1CCOC1)=O 62171,C1(NC(C2CC(C)CN2C(c2ccc(C#N)o2)=O)=O)CC(C)N(C)CC1C 62172,CC(CCN=c1[nH]cnc2cccnc12)NC(=O)CCC1CCCOC1 62173,CC1CCN(C(=O)Cc2cnccn2)C(C)C1NC(=O)CCCC1CCCCC1 62174,N1(C(C(=O)NCC(F)F)C2C(C)C2)CCC(CC(N2CCCCCC2)=O)CC1 62175,C(CC(C(C)(C)C)NC(C1CCC(C)(C)C1)=O)N(C(C1(CCCC)CC1)=O)C 62176,c1(NC(=O)Nc2ccc(C(N(CC)CC)=O)cc2)cc(C)c2c[nH]nc2c1 62177,C(=O)(C(C)C(C)c1ccccc1)NCC(C)NC(CC(=O)OCC)=O 62178,N1(C(C(C(C)C)C)=O)CCN(C(c2ccc([N+](=O)[O-])s2)=O)CC(CO)C1 62179,C#Cc1ccc(C)c(NC(C2CC(C)(NC(=O)CC3CCC(=O)N3C)C2)=O)c1 62180,CC1CN(C)C(C)CC1NC(C1C(NC(=O)COCCF)C1(C)C)=O 62181,c1(C(=O)NCC2CCN(CC)C2)cc(CC2CC2)sc1Br 62182,Cc1[nH]nc(C(N2CCOCC2CN(C(=O)C(F)(F)c2nccn2C)C)=O)c1N 62183,C12(C(=O)NCC3(C(N4CCC(C(=O)OCC)C4)=O)CCCO3)CCN(CC1)CC2 62184,c1(NCCN(N(C)C)CC)ccc(S(=O)(=O)NCCC2CC2)cc1C#N 62185,c1(C(=O)NC2(CC#N)CN(C(=O)CC3CC3)C2)sc(Cl)cc1Cl 62186,c1(C(=O)NC2(C)CCN(c3ncc(C(=O)OC)cn3)C2)cc2n(c1)CCSC2 62187,c1(C(=O)NCC2(CN(C(c3ccc(C)s3)=O)C)CC2)ccc(Cl)nc1N 62188,c1(CCC(=O)NC2CN(C(=O)C(O)CC3CC3)CCC2O)nc2ccccc2o1 62189,C1(NC(CCc2nc(C)sc2)=O)CCC(NC(C2C3COCC23)=O)CC1 62190,C1(C(=O)NC(C#C)C)(NC(=O)C(COC)N(C)C)CC1(C)C 62191,C1(CNC(C(CC)NC(C)=O)=O)CC2CCC1N2C(=O)CCCCN(C)C 62192,C1(NC(c2c(C)ccs2)=O)CC(NC(c2ccc(CC(C)C)nc2)=O)C12CCC2 62193,C1(C(=O)NC2(CCCNC(c3ccc(Cl)c(Cl)c3)=O)CC2)COC2(CCC2)C1 62194,C1(c2nnnn2CC2CCCO2)(NCc2nc(C)sc2)CCCCCC1F 62195,N1(C(C)C)CC(c2nnnn2C2CC2)(NCc2nc(C(F)F)n[nH]2)CCC1=O 62196,C1(C(N(CCNC(=O)C(CCO)N(C)C)CC)=O)CNC(=O)CC1(C)C 62197,C1(CNC(C(F)=CC)=O)CCCC1NC(c1cc(C(=O)NC)[nH]n1)=O 62198,C1(CNC(C(CC)CC)=O)CCN(C(C2CC3CC(=O)C2O3)=O)C12CC2 62199,C(=O)(C(O)C(C)(C)C)NCC(C)(C(C)C)NC(C1(C(N(C(C)C)C)=O)CC1)=O 62200,C(=O)(CCCC(C)C)NCC1CN(C(NOCCC)=O)C(C)C1 62201,c1(SC)ccc(C(=O)NC2CC(NC(=O)CN(C)C(C)=O)C23CCC3)c(Cl)c1 62202,CC(C)(C)CC(=O)OCCC(N1CCC(OC(C)(C)CNC(=O)CON)CC1)=O 62203,C(=O)(NNC(=O)CNc1ccccc1)c1ccc(CN(CC(F)(F)F)C)cc1 62204,N1(C(CCn2c(C)ncc2)=O)CCC2(CCCC2NC(=O)Cc2n[nH]c(=N)s2)C1 62205,CN1CCCC(C)C1.c1(N)cncc(N2CCCC2)n1.n12cc(nn1)CC21CC1 62206,C(=O)(CCCC(C)(C)C#N)Nc1c(OC)cc(NC2CC2)c(Cl)c1 62207,N1(C(CSCC)=O)CC2COCCC2(NC(=O)CC(n2nc(C)cc2C)C)C1 62208,n1(CC(=O)NCC2C3N(C(C(COC)O)=O)C(CC3)C2)nc2ccccn2c1=O 62209,C1(C(=O)NC(C)(C)C=CC(=O)NC(C2CCOC2)(C)C)C2CCC(F)C12 62210,N1(C(c2c(OCC)cccc2)=O)CCC2(CCCN2C(=O)CCc2cccs2)CC1 62211,c1(C(N2CCC(N(C(CCC#CC)=O)CCCC)CC2)=O)cc(NC)ncc1Cl 62212,c1(CC)cc(C(=O)NC2C3CC2N(C(c2oc(C)nc2C)=O)C3)ccc1C 62213,CCC(CNC(=O)CC(C)CN(C)C)(CC)NC(c1ncc(C)cn1)=O 62214,c1(CC)cc(C(=O)NCC(O)CNC(c2cnc(C(C)(C)C)o2)=O)nn1C 62215,N1(C(C(C)CF)=O)CCCC(N2CCN(C(=O)CCc3n[nH]c(=N)s3)CC2)C1 62216,c1(C(N2CC(O)CCC(NC(C(C)N3CCC3)=O)C2)=O)nc2n(c1Cl)CCCC2 62217,c1(C(=O)NC(CNC(C(C)C2CCCC2)=O)(C)CO)cc2c(s1)CC(C)(C)C2 62218,n1(CC)nc(C(=O)NC(C2CCN(C(C3CCCCS3)=O)CC2)C(C)C)cc1C 62219,c1(NC)nc(NC(C2CC(C)(NC(=O)OC(C)(C)C)C2)=O)ccn1 62220,C1(NC(c2c(CC)noc2)=O)CCN(C(c2ccccc2C(C)(C)C)=O)CC1C 62221,N1(C(C(C)CF)=O)CCC(N(c2cccc(C(F)(F)F)c2)C)CC1 62222,c1(C(N2CC(CCC)C(NC(=O)CC(C)OC)C2)=O)cc(C)nc(C)n1 62223,c1(CC(=O)NC(CCNC(CN2C(C)CCC2)=O)(C)C)ccccc1OC(F)F 62224,C(=O)(CCCC(=O)NCCCCNC(c1ccccc1N1CCCC1)=O)OCC 62225,C1(N(C(C(CC=C)CC=C)=O)C)CCCC2CN(C(=O)C(C#N)CCC)CC12 62226,CCN=C(NCCC1(C)CC1(F)F)N1CCc2c(Br)cccc2C1 62227,C1(O)(C(C)NC(=O)CC(C)n2cccn2)CCN(C(c2ccco2)=O)CC1 62228,c1(C(N(CC(C)CO)C)=O)coc(CNC(C2(O)CCOC2)=O)n1 62229,c1(NC)c(C(=O)NC(C2CCN(C(C3CC4CCCC34)=O)C2)C)cccc1N 62230,C(=O)(C(C)CCC(C)(C)C)N1C2CC(C(=O)NC(c3c(C)noc3C)(C)C)C1CC2 62231,C1(C)(CNC(C2N(CC)CC2)=O)CC(OC)CN1C(=O)CC(C)n1cccn1 62232,C1(NC(=O)C(O)Cc2ccccc2)CC2CC1CN(C(C1CCC3(CC3)C1)=O)C2 62233,C12(C(=O)NCCC(C)N(C(c3ccc(C(=O)OC)[nH]3)=O)C)CCCN(CCC1)C2 62234,N1(C(C=C2CCN(C)CC2)=O)CCCN(C(c2ccc(Cl)nc2N)=O)CC1 62235,CN1CC(C)(C(=O)NCC2CC(NC(c3ccn(C4CC4)n3)=O)C2)CC1=O 62236,C1(NC(CCCCSC)=O)COC2(CCN(C(=O)Cn3ccc([N+](=O)[O-])n3)C2)C1 62237,c1(OCC)ccccc1OC(C)C(=O)NC(C)C(C)F 62238,C1(CNC(c2cnc(COC)s2)=O)CCN(c2nnc(O)s2)CC1C 62239,c1(C(C(=O)NCCCCCC)N(C(C#N)C2(COC)CC2)C)cccc2c1CCO2 62240,c1(C(=O)NCC(CC)NC(c2ccon2)=O)ccc(Cc2nc[nH]n2)cc1 62241,Cc1cc(N)cnc1C(N1CC(CC(F)C(=O)NCC(CC)C(C)(F)F)C1)=O 62242,c1(C(=O)NC2CC(NS(=O)(=O)c3cccnc3)C2)cc(Cl)nc(Cl)c1F 62243,c1(NCC(=O)Nc2ccc(C#N)c(I)c2)c(Br)c(O)c(O)c(Br)c1Br 62244,n1(CC(=O)NCc2onc(-c3cccc(C)c3)n2)c(C(C)C)nc2ccccc12 62245,C1(CC)CC(C)CN(C(C2(C)CCCN2Cc2ccc(OC(C)C)cc2)=O)C1 62246,N1(C(c2c(OC)cnc(F)c2)=O)CCCCC(NC(c2ccncc2C)=O)CC1 62247,n1(CCC(=O)NCCCC2(NC(C(C)C#N)=O)CC2)cnc2sccc2c1=O 62248,c1(NC(=O)CC2CN(C(C3CN(C(C)(C)C)CCO3)=O)C2)ncc(Cl)nc1Cl 62249,C1(NC(C(CC)(C)O)=O)COC2(C1)CN(C(=O)C1=CCCOCC1)C2 62250,N1(C(Cc2ccn(C)n2)=O)CC2CC(NC(C3CCCC(C)(C)C3)=O)CC1C2 62251,C1(NC(C=CC(C)NC(c2n(CCC)ncc2)=O)=O)CCN(C)CC1C 62252,N1(C(C2CCCN(CCC)C2)=O)CCN(C(=O)C(C)S(N)(=O)=O)CC(C)(F)C1 62253,c1(C(=O)NC(C(C)NC(COc2c(F)ccc(C)c2)=O)C)cccc2scnc12 62254,c1(C(=O)NCC2N(C(CC3(C=C)CC3)=O)CCCC2C)n[nH]c2c1CSCC2 62255,CC1CCCC(C(N2CC3C(CNC(=O)C=Cc4cnn(C)c4)C3C2)=O)C1 62256,Cc1ccc([N+](=O)[O-])c(C(=O)NCC2CC3CC3N2C(C2CC3CCC2O3)=O)c1 62257,CC1CC(=O)NC(C(=O)NCc2cccc(NC(=O)C(F)(F)c3cncs3)c2)C1 62258,N1(C(C(C)=CC2CC2)=O)CCCCC2(CCN(C(=O)C3=C(C)CCCC3)C2)C1 62259,CC(O)CCN=c1[nH]c(N2CCC(N3CCOC3=O)C2)nc2c1COC2 62260,C1(CNC(=O)CCn2cncn2)CC(F)CN1C(C1CCCCC1)=O 62261,c1(SC)cc(F)ccc1C(=O)NC(C)(C)CNC(c1c(C(F)F)nn(C)c1C)=O 62262,C12(CCN3CCN(C(c4ccc(OC)cn4)=O)CC3)CCC(CC1)C2(C)C 62263,c1(CCC(=O)N(CC(CC)NC(=O)C(C)Cc2cccnc2)C)c(C)noc1C 62264,C1(C(N2CCC(CCNC(CCCC=C)=O)CC2)=O)C(C)(C)CCCC1(C)C 62265,Cc1nc(C(=O)NC2(C(N3CCC(CCF)CC3)=O)CCCC2C)c(C)o1 62266,C1(OC)CCC(CC(=O)NCC2(C)CCCN2C(c2occc2C)=O)CC1 62267,C(C(O)C(F)(F)F)NC(c1cncc(OCCN2CCCCC2)c1)=O 62268,N1(c2n(CCCOC)c(C(O)C(C)OCC)nn2)CCN(C)C(=O)C1 62269,C=CCC(C(=O)N(C1CCN(C(c2ccc(CN(C)C)nc2)=O)CC1)C)C(C)C 62270,c1(C(c2nnnn2C)NC2(CO)CC(OC)C2)ccc(N2CCC2)cc1 62271,N1(C(C2(C)C(C)C2)=O)CC(NC(c2csc(-c3ccco3)n2)=O)C(O)C1 62272,C1(CNC(=O)COc2ccsn2)CN(C(=O)C(c2ccccn2)O)CCCO1 62273,CC1CC2(CCN(C(=O)CCC3CC3)CC2)CN1C(c1ccc(S(C)=O)cc1)=O 62274,C=CC(C)(CCOC)C(=O)NC1CCCCCC1NC(C1CC2(CC2)C1)=O 62275,c1(CNC(CC(=C=C)C)=O)cc2n(n1)CCN(C(c1c(C)cc(Cl)cc1N)=O)C2 62276,CC1(CNC(=O)C(C#N)C2CC2)CCCN1C(c1cnc(S)[nH]1)=O 62277,c1(C(=O)OCC)sc2ccncc2c1NC(=O)CSCc1scc(Br)c1Br 62278,Cc1ccc(C(=O)NC(C)CCN(C(=O)CCc2cnn(C)c2)C)nc1 62279,N1(C(c2ccc(-c3ccco3)[nH]2)=O)CCC2C(CCN2C(C2CCCCS2)=O)C1 62280,C1(NC(CC)=O)(CNC(=O)CNc2nc(C)cs2)CCCCC1C 62281,c1(NC(CC(C)(C)N(C(CC(C=C)C)=O)C)=O)cccc([N+](=O)[O-])c1 62282,C1(C(=O)NCCN(C(=O)C=CCO)CC)CCCC1N(C)C 62283,OCC(F)(F)CCCCN=C(NCc1ccon1)NC1CCC1 62284,Cc1cc(Cl)ncc1NC(=O)C(C)C(C)NC(c1ccn(CO)c1C)=O 62285,C1(C(=O)NCC(C)(C)OCCNC(C=C(C)C(F)F)=O)CC(C2CC2)C1 62286,Cc1cc(NC(c2cncc(N3CCN(C)CC3)c2)=O)c(O)c(C)c1 62287,C=CC(CCC)CC(=O)N1CCN(C(=O)CCc2cccc(O)n2)CC1 62288,Cc1nc(N(C)C)sc1C(N1CCC(C)C1CNC(C12CC(C1)C2)=O)=O 62289,CCCCN=C(NCCc1cccc(F)c1F)NC1CN(C2CC2)C1 62290,C1(CNC(C2(CC#C)CCOC2)=O)CC2CCC1N2C(=O)C(C)(CC)CC 62291,C1(CC(=O)N(CCNC(C(C)OCCC(C)C)=O)C(C)C)CCNC(=O)C1 62292,CCCC(C(=O)OC)C(=O)NCC1(C2(O)CN(C(=O)C=Cc3cnc[nH]3)C2)CC1 62293,c1(N(C)CC2CC=CCC2)nnc(C(F)F)n1CC(=O)OC(C)(C)C 62294,Cc1nc(C=CC(=O)N(C2CCCC2)CCNC(c2cccnc2S)=O)[nH]c1C 62295,c1(C(=O)NC2CC3(CN(C(C=CC=CC)=O)C3)C2)cc2c(OCC)cccc2[nH]1 62296,C#Cc1ccc(F)cc1C(=O)NC1C=CCN(C(c2ccc(F)cc2C#N)=O)C1 62297,N1(C(C(CCC2CC2)NC(C(CC(C)(C)C)O)=O)=O)CCC(C2(O)CC2)CC1 62298,N1(C(=O)Nc2c(COC)cc(F)cc2)CC(C)(C)C(O)C1(C)C 62299,C1(C)(C(=O)NCC(C)(C(C)C)NC(C(CCC)=CCC)=O)CCCCC1(F)F 62300,c1(N(CCCC2N(CCOC)CCC2)Cc2ccccc2)cc(C)c(C#N)cn1 62301,N1(C(C(COC)C)=O)CCC(C(=O)NCC(C)CC2CCC2)(CO)C1 62302,C1(NC(c2c(O)ncc(C(C)C)c2)=O)CCC2CCN(C(=O)C=CCO)C1C2 62303,CCC(CC)C(=O)N(C)CC1CCN(C(c2cnn(CC3CCOCC3)c2)=O)C1 62304,N1(C(C=Cc2occ(C)n2)=O)CC2CN(C(=O)CNC=O)CCC2(CO)C1 62305,C(C1CCC(c2nnnn2C(C)C)(Nc2cccc(F)c2)C1)=CC(=O)OC 62306,C(c1ccc(OC)c(Cl)c1)=CC(=O)NC1CC(C)(CNC(C(CC)COC)=O)C1 62307,c1(CNc2ccc(NC(C3C(C)CCC3)=O)c(F)c2)ccc(C#N)cc1O 62308,C(=O)(N=c1cccn[nH]1)C1CC(C)CN1C(c1ccc(Cl)o1)=O 62309,N1(C(c2ccc(-n3c(SC)ncc3)cc2)=O)CC(C)CC(O)C1 62310,C1(COC2CCCC2)CN(C)CCC1(F)F.c1(CNC(C)C=O)ccn(C)n1 62311,N1(C(C)C)C(=O)NC2CN(Cc3cc(C(C)(C)F)on3)CCC12 62312,N1(C(C(N2CCCCC2=O)C)=O)CC2CCC1C(CNC(=O)CO)C2 62313,N1(C(CC2(OCC)CC2)=O)CCCC1CN(C(=O)Cn1ccnc1C)C 62314,S(=O)(=O)(c1ccc2occc2c1)NC(C(OC)OC)C 62315,N1(C(c2c(COC)n(C)nc2)=O)CCC2(NC(=O)CCCC3CCC3)CC2C1 62316,c1(C2CCN(C(c3[nH]nc(NC(=O)NC4CC4)n3)=O)C2)cc(Br)ccn1 62317,c1(C(N2C(CN(C(c3c(COC)nc[nH]3)=O)C)CCC2)=O)cnc(C(F)F)nc1 62318,C1(CNC(C(C(C)C)OC)=O)CC2CCC1N(C(C13CCCCC1C3)=O)C2 62319,c1(C(=O)NC2CC(NC(c3c(C)nc(CCC)s3)=O)C2)csc2ncnc(O)c12 62320,C(CC(C(=O)OC1CCCC1NC(c1cncs1)=O)NC(=O)OC(C)(C)C)SC 62321,c1(C(=O)NCCCNC(C(C(CC)C)OC)=O)c(Cl)cc(CO)cc1Cl 62322,C(=O)(CCCCC(F)(F)F)NCC12CCC(NC(CC3(C)CCC3)=O)(C1)CO2 62323,CCCC(C(O)C(=O)Nc1ccc(O)c(OC)c1)NC(C1(COC)C=CCC1)=O 62324,n1(CC)c(C)nn(CC(=O)NCCCNC(c2ccc(C(N)=O)cc2)=O)c1=O 62325,C(=O)(C(F)(F)C(F)F)NC1CN(C(c2c(CC)nns2)=O)C(C)C1 62326,CCC(CN1CC(=O)N(CC(C)CSC)C1=O)(CC)C(=O)OC 62327,N#Cc1c(C(=O)OC(C)(C)C)cccc1F.N12CCC3CCCC13COC2=O 62328,Cc1nc2sc(C(N3CC(CNC(=O)C(C)N4CCC4)C3)=O)cn2c1Br 62329,C1(O)(N(C)CCNC(=O)C(C2(O)CN(C(=O)C3CC3)C2)F)CCSCC1 62330,C1(NC(=O)CCC2CC2(F)F)CCN(C(c2ccnnc2O)=O)CC12CCC2 62331,CC(C)CC(CC(=O)NC1(CO)CCC(C)C1)NC(C1CC2(CCC2)C1)=O 62332,c1(C(C)(C)C(=O)NC(CNC(=O)CC2CC=CCC2)CO)ccc2c(c1)OCO2 62333,CC1CCC(CONC(C2CCN(C(=O)C(O)C(C)C)C2)=O)CC1 62334,C1(NC(c2c(C)[nH]nc2CO)=O)CCN(C(c2cc(Cl)ccn2)=O)C(C2CC2)C1 62335,C1(CNC(C2CC(C)C(C)CC2)=O)C(C2CC2)CCN1C(c1cnc(S)n1C)=O 62336,c1(C(N2CC(F)(CNC(C3(OC)CC(CF)C3)=O)C2)=O)cc(Cl)cn1C 62337,N1(C(=O)CCOC2CC2)CCCN(C(C2(C(F)(F)F)CC3CC3C2)=O)CC1 62338,c1(CC(C)N(C(c2ncccc2C)C(=O)NCC)C2CC2)ccc(C)cc1 62339,N1(C(C(C(CC)C)N(C)C)=O)CC2CC(C(N3CCC(O)CC(C)C3)=O)CC2C1 62340,c1(N(CCCC)C)nc2ccccc2c(=NC2CCc3ncccc3C2)[nH]1 62341,N1(C(=O)COc2ccc(-n3cc(Br)cn3)nn2)CC2CCC1CO2 62342,C1(C(=O)OC)C(C)CCCN1Cc1c(-c2cccc(O)c2F)cnn1C 62343,C1(NC(CNC(CNC(=O)OC)=O)C2CCC2)C2CCCCC12 62344,CC(C)S(=O)(=O)C(C)C(=O)NC1(CCNC(c2cc3c(nc2O)CCC3)=O)CC1 62345,c1(C(=O)NC(CN(C(CNC(=O)NC)=O)C)C)cc2oc(Cl)cc2[nH]1 62346,C1(C)(CC(=O)NCC(C(=O)NC(C)Cc2cnn(C)c2)O)CCCCC1 62347,c1(C(=O)NCC(CC=C)NC(c2cc(-c3cccs3)on2)=O)cc(F)ccc1C 62348,C1(CNC(c2ccc(C(C)C)o2)=O)CN(C(C2CCCS2)=O)C2(CCC2)C1 62349,c1(NC(C2(O)CCN(C(=O)CC3COCCO3)C2)=O)cnc(Br)c(Cl)n1 62350,C1(CNC(C2(C3N(C(CNS(CC)(=O)=O)=O)CCC3)CC2)=O)C(C)(C)C1(F)F 62351,c1(N(C(=O)CN(CC(F)(F)F)CCCOC2CNC2)C2CC2)ccc(Cl)cc1 62352,C1(C2CCC2)(CNC(COC2CN(C(C(C)(C)OCCC)=O)C2)=O)CC1 62353,n1(CC(=O)NC2(COC)CN(C(=O)C(C)(C)F)C2)ccc(C)cc1=O 62354,c1(N2CCC(C3(NC(CC(C=C)(C)C)=O)CC3)CC2)cc2c(cn1)C(=O)CCC2 62355,c1(NCCCN(C)C)ncccc1S(=O)(=O)NC1CCCn2nccc21 62356,c1(-c2cn(CC(N3CCC(c4ccc(F)cc4)C3)=O)nn2)cc(F)c(F)c(F)c1 62357,Cc1cc(F)c(C(=O)N(CCCCCCNC(C2COCCN2C)=O)C)cc1F 62358,c1(CNC(C(C)N(C(=O)C(C)C2CCC2)CC)=O)sc(C)cc1C 62359,c1(OCCCOC)cc([N+](=O)[O-])ccc1C(=O)Nc1ccccc1-c1nn[nH]n1 62360,C1(CC)CN(C(=O)CCCC(=O)OC(C)(C)C)CCN1C(C1CCC1OC)=O 62361,c1(OC)ccnc(OC)c1C(N1CC(CNC(c2cn(CC)nn2)=O)C(C)C1)=O 62362,CCC(CC(=O)NCCn1cc(C(=O)Nc2ccc(C)c(O)c2)nn1)C(C)C 62363,N(C1CS(=O)(=O)N(C)c2ccccc21)C(=O)NC(c1cccnc1)CC 62364,Cc1[nH]c2ccccc2c1NC(=O)Cc1ccc(CCC(=O)O)cc1C 62365,CC1(C)CC(C)(C(=O)NC2(CO)CCC2)CN1C(C1CCCOCC1)=O 62366,N1(C(CCCCSC)=O)CC(CNC(=O)C(C(C)(C)C)SC)C2(CC2)C1 62367,Cc1c(Cl)ccc(C(=O)NCC2CCN(Cc3ccnc(Cl)c3)CC2)c1F 62368,c1(C(=O)NC(C)CNC(=O)C(C)n2cncn2)cccc2c1OCCN2C 62369,c1(C(=O)NC2C(CNC(c3ccccc3O)=O)CC2)ccc2nc(CO)[nH]c2c1 62370,C1(NC(C2CCCCO2)=O)CCN(C(=O)Cc2ccccc2Cl)C12CCCC2 62371,C1(C(N2CC(NC(c3c(C)cn(C)n3)=O)C(C)C2)=O)CC2CCC(C1)C2 62372,C(C1c2ccccc2CN1C(=O)OC(C)(C)C)N(C)C(C1(CCO)CN(C)C1)=O 62373,N1(C(C(C)C2CC2)=O)CC(NC(c2cn(C)nn2)=O)C(F)C1 62374,N1(C(C(=O)NCCCF)=O)CCc2nc(S)[nH]c2C1 62375,c1(SC)ncc(C(N2CCN(C(c3cnc(=N)[nH]c3)=O)C(CF)C2)=O)c(O)n1 62376,N1(C(C#CC(C)C)=O)CC2COCCC2(NC(c2nccnc2N)=O)C1 62377,C1(CNC(C(F)=CCC)=O)CC2CCC1N2C(c1cccc(Cl)c1CC)=O 62378,CC(C)C(O)C(=O)N1CC(NC(=O)C=CC2CC2)C(c2ccccc2F)C1 62379,Cc1cc(C(=O)NCC(C)(C)CNC(=O)C(O)Cc2ccc(F)cc2)cc(C)c1 62380,C(=O)(C(C)(C)CCCF)NCC1CC(NC(C(c2n(C)ncc2)O)=O)C1 62381,C1(NC(C(C)OCCOCC)=O)CCN(C(=O)CO)C1 62382,c1(C(N2CCN(C(C(CC#C)O)=O)C(CO)C2)=O)cnc2c(cnn2C)c1O 62383,C1(NC(CNS(CC)(=O)=O)=O)CN(C(=O)C(CC)SC(C)C)Cc2nccn2C1 62384,CC1(CNc2ccc(-n3ncc(C(=O)O)c3C(F)(F)F)cc2)CCC(=O)NC1 62385,c1(NC(C)=O)ccc(C(=O)NCC23CC2CN(C(c2cscc2C)=O)C3)c(Cl)c1 62386,Cc1ccc(C(=O)NCCC(C)NC(c2cnc(C(N)=O)s2)=O)c(N)c1F 62387,CC(CCCCNC(C1CCC(N(C)C)C1)=O)NC(C1CC1c1cnc[nH]1)=O 62388,CCCCS(=O)(=O)CC(=O)N1CCC(NC(c2n[nH]c(CC)c2F)=O)C1(C)C 62389,CC1(NC(=O)CC23CC(C2)C3)CCN(C(c2ccc(N3CCCC3)nc2)=O)C1 62390,C(=O)(C(C)CCC(C)(C)C)NC(CC)(CNC(c1sccc1COC)=O)CC 62391,N1(C(C2CCCN(CCC)C2)=O)CC(CNC(=O)CCc2ccco2)C(C)(C)C1 62392,c1(NC(C23CC(C2)C(C(F)(F)F)O3)=O)ccccc1-n1ccccc1=O 62393,CN=c1nc(N2CCOC(C)CC2)[nH]c(=NCC2(c3cccs3)CCOCC2)[nH]1 62394,c1(OC)cc(C(F)(F)F)ccc1C(=O)NC1(C)CC(NC(=O)Cc2ccon2)C1 62395,Cc1nn(C(C)C)cc1C(=O)NC1(CNC(C2(CF)CC(F)(F)C2)=O)CCC1 62396,C1(C(=O)Nc2ncc(OCC)nc2)CC12CCN(C(=O)CCOC)C2 62397,Cc1nc(=NC(=O)CC2CS(=O)(=O)C2)s[nH]1 62398,Cn1ccnc1C(F)(F)C(=O)NC(CNC(C1(C2CCCO2)CC1)=O)CO 62399,c1(C(=O)NCCN(C(=O)C(C)=C2CC2)CCC)cc(C2CCCO2)n(C)n1 62400,C1(OC)COCC1S(=O)CCCN1CCC(NC(C2CCN(C(=O)OC)CC2)=O)C1 62401,N1(C(c2ccc(C)c(C)c2)=O)CC(C2CN(C(c3cscc3C(F)(F)F)=O)C2)C1 62402,C1(C2CCN(C(C3(CO)CC3(F)F)=O)C2)(NC(Cc2c(C)cc(Cl)nc2)=O)CC1 62403,C1(C(=O)NCc2cccnn2)CSCCN1C(c1ccncn1)=O 62404,c1(CC(=O)NC2(CF)CCN(C(C3(CC#C)CCCO3)=O)C2)ccc2c(c1)CC2 62405,C1(CC(=O)NCC(C)(C2CC2)NC(=O)CCCC2CCCO2)CNC(=O)O1 62406,C1(F)(C(N2CCOCC(NC(=O)Cc3cc(Br)cs3)C2)=O)CCCCC1(F)F 62407,CCC(C)(C)CCCC(=O)N1CCC1C(=O)NCCCC1CCCCO1 62408,CN(C)NC(=O)CCC(=O)NC1(C)CCCCC1C(=O)NCC(F)(F)C(F)F 62409,Cc1cnc(C(=O)NC(CNC(c2cncc(N(C)C)c2)=O)CC(C)C)c(F)c1 62410,Cc1cc(C(N2CCC(NC(=O)Cc3ccco3)C23CC3)=O)cc([N+](=O)[O-])c1Cl 62411,N1(C(C2CCCN(C(=O)OCC)CC2)=O)CC2CCN(C)C2C1 62412,CC1CCC2CN1C(=O)CN2.c1(NC(N)=O)ccccc1.C12(CC1)C(=O)NC2 62413,c1(C(N2CC(S(C)(=O)=O)C2)=O)cccc2ccc(Br)cc12 62414,Cc1ccc(C(F)(F)F)cc1C(N1CC2CC1CC2CNC(=O)CCC#N)=O 62415,C1(NC(=O)CC2CSC2)CCC2CCN(c3ncnc4sccc34)C1C2 62416,O=NN1CCCCC1C(=O)NCc1ccc(CCNC(C2(O)COC2)=O)cc1 62417,N1(C(C2N(C(CC(C)C(F)(F)F)=O)CC(O)CC2)=O)CCC12CCCOCC2 62418,C1(CC=C)(C(=O)NCC(=O)NC2CCC2NC(=O)CCC)CC=CC1 62419,C1(C(N(CCCn2cc(-c3c(C)nccc3)nn2)C)=O)CCn2cncc2C1 62420,C1(OC)CC(C)CN(C(C2CN(C(=O)CC3NC(=O)NC3=O)CCO2)=O)C1 62421,Cc1[nH]c2ccc(Cl)cc2c1C(N1CC(NC(C2CC=CC2)=O)CC(O)C1)=O 62422,N1(C(c2c(OC)nccc2)=O)CCC2CN(C(C3CCCCO3)=O)CC2C1 62423,CCCCC(CC)C(C(=O)Nc1ccc(F)cc1)N1CCCC1C1CCOCC1 62424,Cc1nc(Br)sc1C(=O)NC1CC(CNC(C2CCOC2)=O)C1 62425,C1(O)(CN(C(=O)C(O)CC2CCCC2)C)CCN(C(C2(C)CSC2)=O)C1 62426,N1(C(C2C(C)(NC(CCC(=O)N(C)C)=O)CCCC2)=O)CCOC2(CCCC2)C1 62427,S(=O)(=O)(c1cccc(N=[N+]=[N-])c1)N1CCC(c2c(C#N)cccc2)CC1 62428,C1(C(=O)NC(C(C)(C)C)CNC(=O)C=CSc2ccccc2)CCC2CC1CO2 62429,Cc1nsc2ncc(C(N3CC(CCNC(c4ccoc4)=O)C3)=O)cc12 62430,N1(C(C=CC(C)C)=O)CCC2(CCC2CNC(=O)CCNC(=O)C=CCl)CC1 62431,C1(NC(=O)CCF)CCCN(C(C2(C(=O)NCC3CC3)CCC2)=O)CC1F 62432,C1(CNC(c2ccc(CC)nc2C)=O)CC2COCC2N1C(c1nccn1C)=O 62433,C1(N(C(=O)CC2CC(CNC(=O)C(C)c3ncco3)C2)CCC)CCCCC1 62434,C1(C(=O)NCCc2nc(C(C)C)on2)CC(F)(F)CN1 62435,c1(C(N(CC(CC)NC(c2ccnnc2)=O)C)=O)ccc(C2CC2)o1 62436,C(=O)(C1=CS(=O)CCC1)N(CCC(C(C)C)NC(=O)COc1ccc(F)cc1)C 62437,N1(C(=O)NCCCCl)CC2CC1CN2C(=O)Nc1ncccc1C(F)F 62438,c1(Cn2c(SCCC)nnn2)cc(=O)oc2cc(C)ccc12 62439,C1(C(N2CC(OCCNC(C3CC3(C)C)=O)C2)=O)(CC)CCOC1 62440,C=C(C)C(C)(O)C(=O)NCCN(C(c1ccc(N(C)C(C)=O)cc1)=O)CC 62441,C1(C(N2CCOCC(C(c3ccccc3)=O)C2)=O)NCCOC12CCC2 62442,c1(C(=O)NC(CCNC(C(C)CO)=O)Cc2ccccc2)ncn2cccnc12 62443,CC1(CCC(=O)NCCOc2ccncc2)CN(C(c2cnco2)=O)C1 62444,c1(OC)c(C(=O)NCC(C)(C2CCC2)NC(c2ccc(CO)s2)=O)csc1C 62445,C1(C(N(C(CC)CNC(=O)COCC(C)(C)C)C)=O)CC2(CC2)CO1 62446,C=CCC(CC(=O)NCc1nc(C)cc(O)n1)NC(C12CSCC1C2)=O 62447,Cn1nc(C(N2CCCC(C(=O)NCC34CCC(CC3)OC4)C2)=O)cc1C#N 62448,C1(c2cn(Cc3c(C)cn(C)n3)nn2)CCN(C(=O)CCC(N)=O)C12CC2 62449,C1(C(=O)NC(C)Cn2cccn2)C=CCN(C(C2CCCC(=O)C2)=O)C1 62450,Cc1[nH]nc(C(F)F)c1C(N1CCCC1Cn1cc(CNC(=O)N(C)C)nn1)=O 62451,N1(C(C2(C)COC2)=O)CCN(C(C2CCCC2n2cccc2)=O)C(CC(F)F)C1 62452,c1(CC(N2CCC(N(C)C(c3coc(Br)c3)=O)C2)=O)cccc2nonc12 62453,C(=O)(C1CCCc2nn[nH]c21)N1CCC(CN(C(c2nc(C)nc(O)c2)=O)C)C1 62454,N1(CC(C)C)CCN(C(c2ccc(CC(=O)O)cc2F)=O)CC1=O 62455,C1(CNC(C(C2CN(C(C3(C)C=CCCC3)=O)C2)OC)=O)CCCC(=O)C1 62456,N1(C(COCCOCC)=O)CC2(C1)CN(C(C1CCCS1(=O)=O)=O)CC(C)(C)O2 62457,CCCC(O)CC(=O)N1CCN(C(C2(c3ccccc3)CC2(F)F)=O)CC1 62458,CC(C(F)(F)C(F)(F)F)=CC(=O)NCC1C2CN(c3ccnc(Cl)n3)CC12 62459,C1(C(=O)NCC(C(C)C)O)CN(C(=O)CCS(C)(=O)=O)CC(C)O1 62460,C1(C)(C(N2CC(CCCC)N(C(c3n[nH]cc3F)=O)CC2)=O)CCCNS1(=O)=O 62461,N1(C(CSCC#N)=O)CC(NC(C2CC3CCC2O3)=O)C2CCCCC12 62462,C1(C(N2CC(C)(C)C(c3ccccc3)C2)=O)Cc2ccccc2C(=O)O1 62463,c1(C(=O)NC2C(C(=O)NCCC3(C)OCCO3)C2)ccc(Br)cc1F 62464,c1(OC)cc(NC(=O)CCC(F)F)nc(-c2nc(-c3cccs3)no2)n1 62465,c1(C(=O)NC(CO)C(=O)NCc2ccc3c(c2)CC3)cc2n(n1)CCC2 62466,N1(C(=O)C=C(Cl)Cl)CCCC2(CCN(C(=O)C(F)(F)C3(C(F)(F)F)CCC3)C2)C1 62467,Cc1cc(Cl)c(C(N2CC(NC(=O)CC3CCCN3C(C)C)CC2C)=O)cc1C 62468,C(c1ccccc1)=CC(C(=O)NCCOC1CCN(C(c2occ(C)c2)=O)C1)C 62469,C1(C(=O)NCc2scnc2C)(CC)CCN(C(=O)CC2(O)CCOCC2)C1 62470,N1(C(C)C(=O)Nc2ccc(CC(F)(F)F)cc2)CCC2CCCC12 62471,N1(C(CN(C2CC2)CC)=O)CCCN(C(=O)Nc2cccs2)CC1 62472,C1(C(N2CC(C#C)(C(=O)NCc3ccc(C)c(O)c3)C2)=O)CCC(C)=C(C)C1 62473,CC1CCCC(n2nc(-c3ccoc3)nc2COCC2CC2)C1 62474,Cc1cc(C(=O)NCC(F)CNC(C2CC(C)(C)O2)=O)nc(C)n1 62475,c1(CN(C2CN(C(C)(C)C)C2)CC(F)F)cc2cc(-c3cc(C)cs3)cnc2[nH]1 62476,c1(C(N(C(C)CN(C(=O)C(C)(C)N(C)C)C)C)=O)nn(C)c(Cl)c1Br 62477,c1(CC)cnc(C(N2CCC(C(N3CCC(CCN(C)C)C3)=O)(CC)C2)=O)nc1 62478,CC1(C)C(NC(c2cccc(OC3CC3)c2)=O)CCN1C(=O)C1CC1 62479,CC1C(NC(C2(C)CCNC2=O)=O)CCCN1C(=O)COc1cc(Cl)ccc1Cl 62480,CC1(CNC(=O)Cc2sc(S)nc2C)CCCN1C(=O)C=CC1CCOCC1 62481,C1(CN)CC2CCCC2N1S(=O)(=O)CC1(CCO)CCOC1 62482,C1(C(N(C2CCCC2)CCCNC(Cn2c(C)nnn2)=O)=O)CCOCC1(C)C 62483,c1(C(C)C)ccc(C(N2CCC(O)CC2C(=O)NC(C)CN(C)C)=O)cc1Br 62484,CC(C)(F)CCC(=O)NCCCNC(c1cc(-c2ccc(Cl)cc2)ns1)=O 62485,C(=O)(C(O)C(CCC)NC(c1cc(O)n(C)n1)=O)NCCC(CCC)O 62486,c1(OC)ccc2[nH]c(C(N3CCSC(C(=O)NCC(C)O)C3)=O)cc2c1 62487,N1(C(C2C=CC(NC(c3nc(C)n(C)c3)=O)C2)=O)CC2CC(CO)C(C2)C1 62488,C12(CC1(F)F)COCC(=O)OCC(=O)NC2.C1(F)(OC(=O)CO)CC1 62489,N1(C(C(CCC)C(C)C)=O)CC(NC(=O)C(C)(C)CS(C)(=O)=O)CC12CCCC2 62490,C1(NC(CNC(C(C)(C)C)=O)=O)CCN(C(=O)CN2CCCC2)CC1(C)C 62491,C(=O)(CCC(F)(F)CN=[N+]=[N-])N1CCN(C(c2ncc(C)c(Cl)c2)=O)CC(O)C1 62492,O=C(CCCC(F)(F)F)NC1CC2CC(NC(c3c[nH]c4cccnc34)=O)C2C1 62493,c1(N(CCCCN(C(c2c(CC)nc[nH]2)=O)C)C)nc2ccc([N+](=O)[O-])cc2s1 62494,C1(C(=O)NCC(C)(F)CNC(=O)CC2CCCCCCC2)CCc2nncn2C1 62495,c1(C(NN(CC)C(=O)OCc2ccccc2)=O)nn(C)c2cccnc12 62496,CCCCC1C(=O)N2CCC(F)(C2)C(=O)N1.C(C(C)(C)C(=O)NC)NC 62497,C(=O)(CCCNC(c1cnn(CC2CC2)c1)=O)N1C(CN=[N+]=[N-])CC1 62498,N1(C(C2N(C(C3C(=C)C3)=O)CCC(C)(C)C2)=O)CC2C3CCC(C3)C2C1 62499,Nc1sc2c(c1C(=O)NC1CCCC1NC(=O)C(=C1CCCCC1)F)CCC2 62500,C(=O)(C(C)(CC)OC(=O)CC(=O)N(CC(C)(C)CNCC)CC)NCC 62501,N1(C(c2c(C(C)(C)C)ccs2)=O)CCCCC1c1cn(C2CCCC=C2Br)nn1 62502,Cc1cccc(C)c1C(=O)NCc1ccoc1C(=O)NCC1COCC1N(C)C 62503,C1(C(C)C)(C(=O)NCCN(C(C2C=CCC2)=O)Cc2ccccc2)CCCO1 62504,c1(C(=O)NC2CC(CNC(C3CCC4CC34)=O)C2)ccc(=NCC2CC2)[nH]c1 62505,Cc1cc(N)ccc1C(=O)NCCNC(C1CC2(C1)CC2F)=O 62506,N1(C(c2c(SC)cn(C)n2)=O)CCC(C)(C)C(CNC(=O)C(C)=CC2CC2)C1 62507,c1(C(=O)Nc2ccc(OC(C)C(F)(F)F)cc2)cccc2oc(N(C)C)nc12 62508,N1(C(C(CCF)NC(c2n(CC)ccn2)=O)=O)CCSC(C)(C)C1 62509,C1(NC(c2cc(C3CC3)no2)=O)CCC(CNC(c2ocnc2C2CC2)=O)CC1 62510,c1(C(N(C2CN(C(=O)C3=CCC3)CC2(C)C)C)=O)csc(N=S(C)(=O)CCO)n1 62511,c1(C(N(CCOCCN(C(C(F)OC)=O)C)C)=O)cc(-c2ccc(C)s2)[nH]n1 62512,c1(C(N2CC(NC(CC(CC)OC)=O)C(SC)C2)=O)cc(C)c(N)cc1Cl 62513,c1(OC)cccc(I)c1C(=O)OCCS(=O)(=O)C(F)(F)F 62514,c1(C(N2CCOCC2)C)nc(-c2csc(N3CCOCC3)n2)n(C)n1 62515,C(CCCCCC(=O)N1CC(COC)CC1C)NC(C1CCC(CC)O1)=O 62516,Cc1cc(C(=O)NC2CCCC2(C)CNC(c2cn[nH]c2)=O)c(C)s1 62517,c1(SC(C)C(N2CCN(C(C3(O)COC3)=O)CC2CO)=O)ccc([N+](=O)[O-])cc1 62518,C(CC(C)C)(C(=O)NC)NCC1CCN(c2snc(CC)n2)CC1 62519,C1(CCNC(C=CC)=O)CCCN(C(=O)CC)C1 62520,N1(C(CC2CCN(C)C2=O)=O)CC2CC(NC(=O)CC3(O)CCC3)C1C2 62521,C1(c2c(C(=O)NCC(=O)NC(C)C)c[nH]n2)CCCCN1C(=O)C(C)C1CCC1 62522,C1(NC(C2(NC(CC(CC=C)OC(C)=O)=O)CC2C)=O)CCC(N=[N+]=[N-])CC1 62523,C1(CNC(C2CC(CC(F)F)C2)=O)CC(F)(F)CN1C(=O)CSCC1CCCO1 62524,c1(C(=O)NCC2(F)CC(CNC(c3cc(=O)cc[nH]3)=O)C2)ccc2nccn2n1 62525,CC(C)(C)C(O)C(=O)N1CC(CCNC(=O)C(N)=O)C1 62526,C1(n2c(C(C)C)nc(-c3cccs3)n2)CC2CCC1(C)C2(C)C 62527,C1(N(S(=O)(=O)CC2(OC)CC2)C(C)(C)C)CC(O)C1(C)C 62528,c1(C(=O)NCC(CC)NC(c2nn(C)c(Cl)c2Cl)=O)cc(C)nc2ccccc12 62529,N1(C(c2c(C)nco2)=O)CCOC(C)(CNC(c2cccnc2S)=O)C1 62530,c1(C(c2nnnn2C)NCC(C)CN(C)C)cn(C)nc1OC(F)F 62531,C(C(CC1CC1)C(=O)NCCC1CCCCO1)NC(Cn1c(C)nnn1)=O 62532,C1(C(N(C(C#C)C2CCC2)C)=O)(CC)CCN(C(C2COCCN2C)=O)CC1 62533,C1(C(N(CCCN(C(=O)CCc2nncn2C)C)C)=O)C2CCCCCC12 62534,Cc1cc(CC(=O)NCCNC(c2c[nH]nc2C(F)(F)F)=O)no1 62535,N1(CCCNC(c2c[nH]c(=N)o2)=O)CCN(C(c2ccc(C(N)=O)o2)=O)CC1 62536,C1(CC(C)C)CN(C(=O)CC2(CNC(C3CCN3C(C)(C)C)=O)CC2)CCO1 62537,C(C)(C(C(=O)NCCCCCN=[N+]=[N-])C(C)C)NC(C(CSC)OC)=O 62538,c1(C(N2CCC(C(C)NC(=O)CC3(C#N)CC3)C2)=O)ccc2c(c1)CC2 62539,C1(C(N2CCC(C(CNC(CSC)=O)(C)O)CC2)=O)CCCCN(C)C1=O 62540,C12(NC(CC3CCC(C)C3)=O)CCC(C(=O)NCC(C)(O)C3CCC3)(CC1)C2 62541,N1(C(C(C)Cn2cccn2)=O)C2CCC1CC(NC(c1cnn(C)c1F)=O)C2 62542,Cc1ccc(Br)c(CN2CC(NC(c3cnc(O)c(Br)c3)=O)C3(CC3)C2)c1F 62543,C1(OCC(=O)NCCN2CCN(C(C3CC3(F)Cl)=O)CC2)CCC(F)(F)CC1 62544,C1(NC(C2(C)COC2)=O)CCN(C(=O)CSc2ccncc2F)CC1(C)C 62545,Cc1cccc(C(CNC(c2cocn2)=O)NC(=O)CC23CCCC2C3)c1 62546,CCC(C)CC(C)C(=O)NCC1(C(N)=O)CN(C(c2ccc(OC)c(Cl)n2)=O)C1 62547,N(C1c2ccccc2CC12CCCC2)C(=O)NC(CSC)Cc1cccc(Br)c1 62548,C1(NC(c2cc(CCC)oc2C)=O)CCCN(C(c2nc(CC)oc2C)=O)C1C 62549,c1(CNC2C(CC3(c4c(Br)ccc(C)c4)CC3)CCC2)ccc2c(c1)OCCO2 62550,N1(CC(=O)NCC(CNC(=O)CCc2n[nH]c(=N)s2)OC)CCS(=O)(=O)CC1 62551,Cc1ccc(-c2cnc(NC(=O)NC(CC3CCOCC3)CO)s2)cc1Cl 62552,c12ncccc1OCc1ccc-2s1.C1(NS(CC)(=O)=O)CCCNC1 62553,C1(CNC(C2CC(C)SCC2)=O)CN(C)CCN1C(c1cccnc1N)=O 62554,C1(C)(C(N(CC(O)CO)C)=O)CCCN(C(=O)CC2NC(=O)NC2=O)C1 62555,c1(C(=O)NC(C(=O)NCC=C=C)Cn2cncn2)cc(O)ncn1 62556,CC1CN(C(=O)C(O)CC(N)=O)CCC1C(=O)NCCC1CCCC1O 62557,C(=O)(C(C)C(F)(F)F)N1CCC(CC=C)(NC(c2cn(CC3CCCO3)nn2)=O)C1 62558,C(=O)(C1=CCC(C)CC1)N1CCC(CCNC(C2CCCC(OC)C2)=O)CC1 62559,c1(CC)nc(C(=O)NC(C2CN(C(c3cnn[nH]3)=O)C2)C)n[nH]1 62560,C1(OC)CCC12CC(C(=O)N(C)CCN(C)C(C1CC3CCC1O3)=O)C2 62561,c1(C(=O)N(c2cnn(C3CNC3)c2)Cc2c(F)cc(F)cc2Br)cccc([N+](=O)[O-])c1 62562,n1(CCCOC)cc(CCC2CN(C(=O)CC(C)C3CCCO3)C2)nn1 62563,c1(CC(=O)NCC2(NC(C(C)n3cccn3)=O)CCCC2)cccc(C(F)F)c1 62564,Cc1[nH]c(C(=O)NCC2CN(C(C3CN(C)CCO3)=O)CCCO2)c(C)c1C 62565,Cc1csc(=NCC(=O)NCC2CC(C)N(C(c3cscc3F)=O)C2)[nH]1 62566,C1(NC(C(C)(C(C)C)OC)=O)CCC2(CCCN2C(=O)CS(=O)(=O)C2CC2)CC1 62567,CC1CCC(C(=O)NC(c2ncccn2)C)N1C(C12CC(C(=O)O)(C1)C2)=O 62568,C#CCC(C)(CNC(=O)C(CNC(=O)C(C)NC(=O)OC)CC=C)CO 62569,C1(CCC)CCCC1C(=O)N(C(C)CCNC(=O)C(C)OCc1ccccc1)C 62570,C1(NC(c2csc(CC(F)(F)F)n2)=O)CCN(C(c2cc(Cl)cnn2)=O)C12CC2 62571,c1(OC)ccc(C(=O)NCC2CCCCC2NC(c2n[nH]cc2F)=O)cc1F 62572,Cc1cnc(NCC2CCCN2C(C2Cc3cscc3C2)=O)nc1S(C)(=O)=O 62573,N1(C(CC2(N(C)C)CCC2)=O)CC(C)(C)CC1CC(N1CCCC(C(F)F)C1)=O 62574,Cc1noc(Cl)c1CC(=O)NC1CCN(C(=O)CC2C=CS(=O)(=O)C2)C1C 62575,N#Cc1ccc(CN2CCC(CC(=O)NCC=Cc3cccnc3)C2)c(Cl)c1 62576,N1(C(CC(CC)CC)=O)CC=C(CC(=O)Nc2c(C)nn(C)c2C(N)=O)CC1 62577,O=C1CC2(C1)CC(C(=O)NCC(CC1CC1)C(=O)NCC(F)CO)C2 62578,CC1CC2(CO1)CN(C(C1(CCNC(=O)C(C)(C)C)CCCC1)=O)C2 62579,C1(CNC(=O)C(=O)NCC23CC(F)(C2)C3)CCCCS1 62580,c1(C(=O)NC(CC=C)CNC(C2CCCC23CCC3)=O)ccnc2c1cnn2C 62581,N1(C(C)=O)CCC(C(=O)Nc2oc(C)nc2SCC2CCCCO2)C(C)C1 62582,C12(NC(c3c(F)ccc(C)c3)=O)CC(C)(C1)OC21CN(C(=O)CC(C)C)C1 62583,Cc1cc(CNC(=O)CCN(C(=O)CC2CCC3CC23)CCO)sn1 62584,N1(C(C(C2CCN(C(Cn3nc(C)oc3=O)=O)C2)(C)C)=O)CC(C)OCC1C 62585,N1(C(C2(C)CCCS2)=O)CCC2(CCC2NC(c2cnc[nH]2)=O)CC1 62586,C(=O)(CC1=CCCC1)NCCC1(NC(CCc2c(C)noc2C)=O)CCOCC1 62587,C1(NC(c2cn(C)c(=O)cn2)=O)CCCC12CN(C(=O)CC1CC(C)(C)CO1)C2 62588,Cc1cc(=O)oc(C)c1C(=O)NC1CCC(F)(CNC(=O)C2=CC3CCC2C3)C1 62589,c1(C(=O)NCC23CC2CN(C(=O)CCCc2nccs2)C3)ncc2ccccn12 62590,N1(C(C(COC)C)=O)CC(NC(c2[nH]nc(C(F)(F)F)c2C)=O)C(O)C1 62591,c1(C(=O)NCC2(OC)CCN(C(CC)=O)C2)nn(C)c(=O)n1C 62592,c1(C(=O)NCC(C2CC2)NC(c2cccc3oncc23)=O)coc2c1COC2 62593,CCC(C)(CC(=O)NCC=CCNC(c1ccc(S(C)=O)cc1)=O)C(=O)OC 62594,N1(C(CN(C2CCC2)C)=O)CCCC(C2(NC(c3cc4c(s3)CCCC4)=O)CC2)C1 62595,Cc1[nH]nc2ncnc(N3CCC(NC(=O)CCC(N)=O)C3C)c12 62596,c1(CNC(=O)NCC2(Cl)C(C(C)(C)C)C2)ccc2c(c1)NCCC2=O 62597,C(CC(N)=O)(C(=O)NCc1cccs1)NC(CC(CN(C)C)O)=O 62598,N1(C(C(=O)NC(C(CC)n2cccn2)=O)OC)CCN(c2nccs2)CC1 62599,C1(CN(C)C(C2CCCCC2)=O)CCCN1C(=O)CCCc1nccs1 62600,c1(C(=O)NC2CCCC(NC(C3CCC(F)(F)C3)=O)C2)cc(F)ccc1C1CC1 62601,N1(C(CCOC)=O)CCC2(CC1)CCN(C(=O)C(C)CCC(C)(C)C)C2 62602,C1(=O)C(F)CC(C)(C)N1.CC(C)C(C)(O)CN1CC(N2CCNC2=O)C1 62603,Cc1ccc(C(=O)NC2C(C(=O)NCC3CC(=O)N(C)C3)C2(C)C)cc1F 62604,C1(C(=O)NC2C(c3cc(F)cc(F)c3)(C)C2)CCS(=O)(=O)C12CCC2 62605,n1(-c2c(Cl)cccc2)ncc2c1CCCC2CN1Cc2cc(O)nnc2C1.C1(C)CCCO1 62606,C1(C(=O)NCC(COC)NC(C2CC=CCC2C)=O)CCCCC12CCC2 62607,CCCCC(C(=O)NCCC(C)C(C)C)NC(C1CCO1)=O 62608,c1(C(=O)NC2CC(C)(CNC(C3(c4ccncc4)CC3)=O)C2)ccc(O)nn1 62609,O=[N+]([O-])c1ccc(Oc2nc(-c3n[nH]cc3Br)n(C3CC4CCC3CC4)n2)cc1 62610,c1(C(N2CCC(CN(C(C(CC#C)O)=O)C)CC2)=O)cccn2nnnc12 62611,CC(c1ccsc1)=CC(=O)NC(C)(C)C(C)NC(=O)CC(C)n1cccn1 62612,c1(COC)nc2cccc(C(N3CCSCC3C(=O)O)=O)c2[nH]1 62613,c1(C(=O)NCC(=C)CCNC(=O)C(F)C2CCOC2)nn(CC)cc1[N+](=O)[O-] 62614,Cc1cc(F)ccc1NC(=O)C(=O)NC(c1ccccc1F)C 62615,c1(C(=O)OC(C)C(=O)Nc2ccc(N(C)C)cc2)cc(Br)c2occc2c1 62616,N1(C(C(CC)N(C)C)=O)CC2CC2(CNC(c2nn(CC)nc2Br)=O)C1 62617,c1(CC)cc(C(N2CCCC2CNC(=O)Cc2cc(C)[nH]n2)=O)ns1 62618,c1(C(N(CCC(=O)NC(CC)C(=O)NC)CCCO)=O)cnc(O)c(F)c1 62619,CC1CN(C(C2CC(n3cc(C45CCC(CC4)C5)nn3)C2)=O)CC1CC(F)(F)F 62620,c1(C2(NC(CC=C=C)=O)CCC2)ccc(CNC(c2cnn(C(F)F)c2)=O)cc1 62621,C1(NC(c2c(C)c[nH]n2)=O)CCC2(CC1)CN(C(C1CC3(C)CCC1(C)O3)=O)C2 62622,C(C(F)C(=O)NCc1cc(C(C)C)no1)C1CN(C(C(C)N(C(C)=O)C)=O)C1 62623,c1(C(=O)NCC(CNC(C2(CC)CCNC2=O)=O)(C)F)n[nH]c2c1COCC2 62624,N1(C(C(CC=CC)C)=O)CC(NC(c2ccnn2C)=O)C2(CCC2)C1 62625,C1(CNC(C(CC)C)=O)CC(O)C(O)CC1C(=O)N(CC)Cc1ccoc1 62626,Cc1ccccc1-c1cc(NC(=O)NCCC#N)on1 62627,Cc1c(CNC2=NCCC2)cc(-c2ccccc2)n1C1CCCCCC1 62628,c1(OC)cc(C)ccc1CNC(=O)CN(C(=O)C1=CCCC1)C(=O)C(C)C 62629,Cc1ccc([N+](=O)[O-])c(C(=O)O)c1.C1C(=O)NOCC(=O)N1CCO 62630,C1(CNC(C2(SCC)CC2)=O)CCN(C(C2C=CCC2)=O)CC1C 62631,c1(CC)ccc(C(=O)NC2(C)CCN(C(c3c(OC)nsc3OC)=O)C2)nc1 62632,N1(C(C2N=C(C)SC2)=O)CCN(C)C(CNC(=O)C=Cc2ccccc2F)C1 62633,C1(C(N(C(C)CCNC(=O)Cc2sccc2Cl)C)=O)CCCCC1O 62634,C1(NC(C2(NC(c3c(CCC)cccc3)=O)CC2)=O)CN(C)CC12CC2 62635,O=S(=O)(c1ccccc1S(=O)(=O)NC1CCN(Cc2ccccn2)C1)C(F)F 62636,c1(C(=O)NC2C(NC(c3nc(C(=O)OC)sc3)=O)CC2)ccc2cncn2c1C 62637,N1(C(c2cccc(C)c2)C(=O)NCCCC)CC(O)CC2(CCCC2)C1 62638,C1(NC(C=CC(C)(C)NC(C(CSC)O)=O)=O)CCCCC12CC2 62639,c1(OC)cc(OC)nc(C(N2C3CCC2C(CNC(=O)CC2=CCCC2)C3)=O)n1 62640,c1(C(=O)NCC(C)N(C(c2ccc(OC)cc2)=O)CC)cccc2nncn12 62641,c1(C(=O)NCC(CCOC)NC(c2[nH]c(O)nc2C)=O)cc2occc2[nH]1 62642,C1(C(=O)NCc2c(C)cccc2)CCC(C)(C)N(C(C2CCCCCCC2)=O)C1 62643,C1(NC(CCS(N)(=O)=O)=O)CC12CCN(C(C1CCC1c1nc[nH]n1)=O)CC2 62644,CCC(CC(F)F)C(=O)NC(C1CCN(C(=O)Cn2cc(C)cn2)CC1)(C)C 62645,CCCCCC(C(=O)NCCC1CN(C(=O)C=Cc2ncc[nH]2)CC1C)C(C)C 62646,C1(OCC(=O)NCC2(F)CCN(C(CNC=O)=O)C2)CCC(F)(F)CC1 62647,c1(CC)cc(C)c(C(N2CCC(CN(C(=O)Cc3csc(Cl)n3)C)C2)=O)o1 62648,Cn1nc(Br)cc1C(c1nnnn1C1CCC1)NCCCOC1CCOC1 62649,c1(C(CC(=O)NCCCOC)NC(c2nccn2C)=O)ccc(C#N)cc1 62650,CC1CN(C(c2cnn(CC(F)(F)F)n2)C(=O)NCCC2CC2)CC2(CCC2)O1 62651,c1(NC(C2CC(O)(CNC(C3CC3c3ccccc3)=O)C2)=O)ccc(O)c(Cl)c1 62652,C(N=c1nc(N2CCC(COC)CC2)c2[nH]ccc2[nH]1)C1(CC)CC1 62653,C1(C(C#C)C)CCN(C(C2(CC)CCCN2C(=O)Cc2nnc(S)n2C)=O)CC1 62654,C(=O)(CCC(=O)NN(C)C)NCCC(C)NC(c1nccc(COC)c1)=O 62655,C1(O)(CN(C(CSC)=O)C)CCCN(C(=O)C(C)(C)OC)C1 62656,c1(C(C(=O)NCCC)N(CC(C)S(C)(=O)=O)C)snc(OC)c1Cl 62657,C1(NC(C(C(C)C)OC)=O)CCN(C(=O)CC(C)(O)C2CC2)CC1(C)C 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62747,c1(C(=O)OC)cc(=NCC2CCCCC2NC(c2cc(Br)ccc2Cl)=O)[nH]cn1 62748,Cc1ccc(Cl)c(C(N2CCC(CCNC(C3CCCCO3)=O)C2)=O)c1N 62749,C1(C2CCN(C(c3ccc4cncn4c3)=O)C2)(NC(CC(C=C)C)=O)CC1 62750,C1(O)(CCNC(C2(CC)CC2)=O)CCN(C(=O)CN2CCCC2C)CC1 62751,c1(N2CC(CO)OCC2)[nH]c(=NCCC(O)C2CC2)nc2sccc12 62752,C1(CNC(c2nccc(CC)c2)=O)COC(C)(C)CN1C(C1CC(F)C1)=O 62753,Cc1cc(C(=O)NCC(O)CNC(=O)C(C)n2cccn2)c2c(n1)CCCC2=O 62754,C1(CCNC(Cc2c(C)n[nH]c2)=O)CN(C(=O)CCCC(=O)N(C)C)CC(C)O1 62755,C1(C(=O)NCCC(C)(C)NC(c2cc(CC)nn2C)=O)CC2(CCC2)CO1 62756,c1(C(N2CC3C(C(=O)NCC(CSC)(C)C)C3C2)=O)cc2n(n1)CCC2 62757,C(=O)(C(F)C(C)C)NC(C1N(C(c2nc(C(=O)NCC(=C)C)sc2)=O)CCC1)C 62758,CC1CCc2onc(C(=O)NCC(C)(C(=O)O)c3ccc(F)cc3)c2C1 62759,c1(CC(=O)NC2CC(N(C)C(c3cnc(O)n3C)=O)C2)cnn2c1OCCC2 62760,CCC(CC)(CCNC(C1CC2(CCO1)CC2)=O)NC(C1C(C)(C)C1(F)F)=O 62761,S(=O)(=O)(c1ccncc1)NC1CCC(NC(c2ccccc2Cl)=O)C1 62762,C1(C#N)(N)CCNC1.c1(SC)ccccc1CC(c1ccnn1C)=O 62763,C1(CNC(c2nc(C)sc2)=O)CC2(C1)CN(C(=O)CC1CCCOC1)C2 62764,N1(C(C(=O)NC)=O)CCCCC1C(=O)NCCOCC(F)F 62765,c1(C(=O)NCC2OCCN(C(C(CCC)C)=O)C2)c(C)nn(C)c1-n1cccn1 62766,N1(C(C(C)Nc2nnnn2C)=O)CCC(C(=O)OC2CN(C(N)=O)C2)CC1 62767,C1(NC(c2cc(C(C)C)no2)=O)CC(F)CN(C(c2ccc(CO)c(Cl)c2)=O)C1 62768,c1(C(=O)NCCSCC(=O)N(C(CC)C2CC2)C)ccncc1Cl 62769,C(CCN(C)C)(C(=O)NC(C)CCCCO)NC(Cc1ccc(C)s1)=O 62770,N1(C(CC(C)OC)=O)CCC2(CC1)CC(NC(=O)C=C(C)C(C)C)C2 62771,N1(C(C2N(C(c3ccc(C)s3)=O)C(C3CC3)CC2)=O)CC2(CCOCC2)C1 62772,C(=O)(C1CCCc2nc[nH]c21)NCCCNC(c1c(C)n(C2CC2)cc1)=O 62773,c1(OCC)cnc(C(=O)NCCC2CN(C(=O)C(C)COC)CCO2)cn1 62774,CC1CCCCN1CC(=O)NCCCCNC(c1cccc(C(=O)C2CC2)c1)=O 62775,N1(C(C(CC=CC)C)=O)CCN(C(=O)COc2ccc(SC)cc2)CC1C(C)C 62776,Cc1nc(O)nc(S)c1C(=O)N(CC(C)CNC(C1CSC1)=O)C 62777,c1(C(N(CCNC(C(C)NC(CC)(C)C)=O)C(C)C)=O)sccc1Br 62778,c1(OC)ncc(C(=O)NCC(n2cc(-c3ccccc3N)nn2)C)c(C)c1Br 62779,c1(C(N(CC(=O)N(CC(=O)N(C)C)C)CC)=O)ccc(C#N)n1C 62780,N1(C(C2(OCC)CCOC2)=O)C2CCC(C2)C1C(=O)NCc1csnc1C 62781,CC(C(=O)NN1CCCC1C(=O)N(C(CO)CO)C(C)C)=CC1CC1 62782,Cc1cc(C(=O)NC2CS(=O)(=O)CC2NC(=O)C(C)N2CCCC2)cc(C)n1 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63135,C1(CNC(CCOCCOC)=O)CC2(CN1C(=O)CCC1(C)CC1)CC2(F)F 63136,c1(CC(C)C)cc(C(=O)NC2CCCC2NC(c2ccc(Cl)o2)=O)n(C)n1 63137,C#CC1(N(C)C)CCN(C(C(=O)NC2CCOC2)c2ccoc2)CC1 63138,c1(C(N2CC3C(N(C(c4cn(CC)nc4C)=O)C)C3C2)=O)c(F)cc(N)cc1F 63139,c1(C(N2C(CNC(C(=O)N(C)C)=O)C(C)(C)CC2)=O)cc2ccc(Cl)cc2o1 63140,c1(C(=O)NCC23N(C(c4c(C)nccn4)=O)CCC2CC3)cc(F)c(Cl)cc1F 63141,C1(C(N2CCC(C(C)(C)NC(c3c(C)noc3C)=O)C2)=O)CC2(COCCO2)C1 63142,C1(CNC(=NCC=C)NC(C)CC)CS(=O)(=O)c2ccccc2O1 63143,c1(C(=O)NC(CCCNC(c2c(CC)con2)=O)C)cc(O)c2ccccc2c1 63144,N1(C(CCCCOC)=O)CCCCC2(C1)CN(C(c1[nH]c(C)nc1C)=O)C2 63145,c1(C(=O)NCC2(F)CC(NC(CC3N(CC)CCC3)=O)C2)ccc(OC)cc1 63146,c1(C(N2CCc3nc[nH]c3C2)=O)cn2cc(-c3cccc4ccoc34)ccc2n1 63147,c1(C(=O)OC)nn(C)c(CC)c1N=c1cc[nH]c(C2CC2)n1 63148,CCCCCCC(C)CC(=O)NC(CNC(=O)C(=O)NC(C)C)C1CCC1 63149,c1(C(N2CCN(C(C(COC)C)=O)C(C)C2)=O)cc2c(Br)cccc2c(=O)o1 63150,C1(CC)(NC(=O)C(C(C)O)c2ccccc2)CCN(C(=O)CN(C)C2CC2)CC1 63151,C(=O)(C(CC(C)(C)C)OCC)NCC1(F)CCC(NC(CCSCCC)=O)CC1 63152,C1(CNC(c2c(C)sc(Cl)n2)=O)CN(C(c2n[nH]cc2C2CCC2)=O)CCN1C 63153,N12CCC(C(F)(F)CC1)CNC(=O)Oc1c(OC)ccnc1C2=O.C(C)(C)(C)OC 63154,c1(CC)cc(C(=O)NCC(C)CN(C(=O)CC2CCCN2CC)C)cc(Cl)c1 63155,C1(C(=O)Nc2cn(CCC#C)nc2)CCCN(C(=O)C(C)=C2CCCC2)C1 63156,C(CNC(=O)CNS(=O)(=O)NC)(CCCC)NC(C1(C#C)CCC1)=O 63157,N=c1nc(N2CC3CCCCC3C2)[nH]c(=NCC2CC(c3ccccc3F)C2)[nH]1 63158,N1(C(C(CC(C)C)O)=O)CC(CNC(c2nc(=N)cc[nH]2)=O)CC12CCOCC2 63159,c1(N2CCCC(CNC(C3(C)CS(=O)(=O)C3)=O)C2)ncccc1[N+](=O)[O-] 63160,c1(C(N2CCN(C(=O)C(O)CN(C)C)C(CCO)C2)=O)c(F)cccc1F 63161,C12CCCC1C(=O)NC2.C1(CC(=O)NCCCCc2cnc[nH]2)(N(C)C)CCC1 63162,c1(CNC(C2C(NC(CNc3ccc(C)cc3)=O)COC2)=O)cc(F)ccc1F 63163,c1(C(=O)NCC2CC(NC(C(C3CCCC3)OCC)=O)C2)ccn2nncc2c1 63164,c1(C(=O)NC2(C)CN(C(=O)C(C)(C)c3ccns3)C2)scc(Cl)c1Cl 63165,c1(C(=O)NC2C(C)CN(C(=O)CCC(F)F)C2)n[nH]c2c1CC(C(C)(C)C)CC2 63166,C(=O)(C(C)C(C)(C)c1ccccc1)NC(CNC(c1c(C)c[nH]n1)=O)CC(C)C 63167,C1(C(=O)NCC(CCC)O)CC(NC(=O)CCC2(C)N=N2)C(O)C1 63168,C1(C(N2CC(C)C=C(C)C2)=O)COC2(C1)CN(C(C1CC3CCC(C1)O3)=O)C2 63169,Cn1cc2cc(C(=O)NCCC(C)(C)CNC(c3c[nH]c(=N)o3)=O)ccc2n1 63170,C1(CNC(COCCC=C)=O)C2CCC(C2)N1C(c1cccc(OC(C)=O)c1)=O 63171,c1(C(=O)NCCOC2CCN(C(C(COC)(C)O)=O)C2)cc(Cl)c(C)cn1 63172,C(=O)(CC1COc2ccccc21)NCCN(CC(=O)NC(c1ccc(F)cc1)C)C 63173,c1(C(=O)NCC(=C)CCNC(=O)C(CC)NC(C)=O)cc2sccc2s1 63174,C1(C(N2CC(CC(=O)NC(C=C)C3CC3)(OC)C2)=O)CCCC(O)C1 63175,c1(OC(N2CC3C(C(=O)OCC)C3C2)=O)c(Cl)nnc(Cl)c1Cl 63176,C#CCCCCCC(=O)N(C1CCCN(C(=O)Cc2ccc(O)cc2)C1)C 63177,c1(NCCCN2C(C)CCC2)nc(N2CCC(CSC)C2)nc2c1ncn2C 63178,N1(C(CC(CC)OC)=O)CC(NC(=O)C(c2ccccn2)C)CC12CCOCC2 63179,N1(C(c2c[nH]c(=N)o2)=O)CCC2(C1)CN(C(c1cscc1Br)=O)CCO2 63180,N#Cc1c[nH]c(C(=O)NC2CN(C(=O)CC3CCC(C4CC4)O3)CC2CO)c1 63181,Cc1ccc(C=CC(=O)NCCN(C)C(C2CN(c3nnnn3C)C2)=O)o1 63182,N1(C(C(C(C)C)OC)=O)CC(C(=O)NCCc2ncccc2F)C(C2CC2)C1 63183,N1(C(CC(CC)(F)F)=O)CC2CCCCC2(CNC(=O)CCc2cnc[nH]2)C1 63184,CON(CCC(=O)NCC1CC2CCC1O2)C(=O)c1cccc2ccoc12 63185,C1(C(=O)OC)C2CCC(C2)N1C(=O)CCn1cc(CC2CCOC2=O)nn1 63186,Cc1ccc(C=CC(N2CCC(C(O)CNC(c3cnc[nH]3)=O)CC2)=O)o1 63187,C(CCCCC(=O)NCC1=CCCC1)N(C(=O)C(F)CC1CCOC1)C 63188,CCCC(C)(C)CC(=O)NC1CC=C(C(=O)N2CC(C3CC3)OC(C)C2)C1 63189,CCCCC(C)(F)C(=O)NCc1nc(C(=O)NCc2cccnc2C)co1 63190,C(C)(C(=O)N(O)Cc1cn(C2CCCC2O)nn1)Oc1ccc(C)cc1 63191,c1(CNC(CCC2CC(NC(CCN(C)CC)=O)C2)=O)nc(C)sc1C 63192,N1(C(c2c(C)nc(Br)cc2)=O)CC2(CCN(Cc3cccc4[nH]ccc34)CC2)C1 63193,N1(C(C(C)Sc2nccn2C)=O)CCCC(O)(C(C)NC(c2cnn(C)n2)=O)C1 63194,C(=O)(CCCC(C)=O)N1CC(CCNC(CCCc2cc(C)no2)=O)C(C)C1 63195,Cc1ccc(F)c(C(=O)NC2CC(c3ccccc3)(NC(c3cc[nH]n3)=O)C2)c1 63196,c1(OC)cnc(C(N2CCCC2CNC(=O)CC(C)O)=O)c(F)c1 63197,CCC(C)(C)C(O)C(=O)N1CC(CNC(=O)Cn2ncc(C#N)c2N)C(C)(C)C1 63198,c1(OCC)cc(C(=O)NCC(C2CC2)N(C)C(c2ccsc2C)=O)ccc1C 63199,N1(C(C2(COC)CC=CCC2)=O)CCCC(NC(=O)COC)CC1 63200,c1(OC)ccc2c(n1)NC(C(N1CC(C(C)NC(=O)CC=CC(C)(C)C)C1)=O)C2 63201,C12(C(=O)NCCN(C)C(c3sc(N(C)C)nc3Cl)=O)CCC(F)(CC1)CC2 63202,c1(C(=O)NC2C(NC(CCNC(=O)C=CCl)=O)CCC2)nccc(Cl)c1Cl 63203,c1(OC)ccc(CCC(N2CC(F)(CNC(=O)C=C(C)C(C)C)C2)=O)cn1 63204,C1(CC(C)C)CN(C)CCN1C(=O)NC1CCC(O)C(C)C1 63205,c1(OC)ccccc1CC(C(=O)O)NC1CCC1.C(C)(=O)OC 63206,c1(N2CCC(C(CCc3ccccc3)NC(C(C)N(C)C)=O)C2)ncccc1C#N 63207,N1(C(CCCC)=O)CC2ON=C(CNC(c3cn(-c4cncc(F)c4)nn3)=O)C2C1 63208,C1(NC(c2cc(C(C)=O)oc2)=O)CC2CC(C1)N(C(C1CC=CCC1)=O)C2 63209,O=C(C(F)C(F)(F)F)NC1CC2(C1)CN(C(=O)CCc1ccc(Cl)cc1)C2 63210,N1(C(c2ccc(C)nc2C)=O)CC2CCCC2(C(N2CCCCCC2CO)=O)C1 63211,N1(C(C(C)(C2(C)CC2)OC)=O)CC2C(CNC(C3CCC=CCC3)=O)C2C1 63212,CC1N(C(=O)C(C2CCNCC2)F)CCCC1(C)C 63213,c1(SC)ncc(Br)c(=NC2CC(C(N3CCN4C(=O)OCCC4C3)=O)C2)[nH]1 63214,N1(C(c2c(C)coc2)=O)CCC2(CC2)CC1C(=O)NC1CC2(CCC2)C1O 63215,Cc1cnc(C(=O)NC2(C)CCCN(C(C3CCOC(=O)CC3)=O)C2)c(Br)c1 63216,C1(OC)CC(NC(c2cccc(CO)c2)=O)C12CCN(C(=O)CSC(C)C)CC2 63217,C1(c2cn(CC3N(C(CN(CCOC)C)=O)CC=C3)nn2)(OC)CCCC1 63218,N#Cc1cccc(C#N)c1N1CCC12CCCOC2 63219,O=C(C1=CC2C=CC(C1)C2)NCCCC(O)C(=O)NCCCC(F)F 63220,Cc1cncc(C)c1C(=O)NCC(O)CNC(=O)C(c1ccccc1)F 63221,C12(CNC(C3C(C)CC3)=O)CCC(CC1)N(C(c1cnn3ncccc13)=O)C2 63222,C(CNC(c1cnc(Br)s1)=O)(CC(C)C)NC(CN(CC)CC)=O 63223,C1(C)(C(N2CCC(C(=O)NCC(=O)N(C)CC)CC2)=O)CCC2CC2C1 63224,C(CCC)(C(=O)NC(C)(CNC(c1c(C)n[nH]c1C)=O)C1CC1)=CCC 63225,c1(C(=O)NC2(CNC(C(C)(C)OC)=O)CCCCC2C)nnc2ccccn12 63226,c1(CC)c(C(N2CC3CC3C2C(N2CCOC(C)C2)=O)=O)ccn1C 63227,c1(NC(C(CCOCC)NC(C2(CCOCC)CCC2)=O)=O)c(C#N)cnn1C 63228,N1(C(CN(C(C)C)C)=O)CCN(C2CN(C(C3CC34CCC4)=O)C2)CC1 63229,N1(C(C(C(CC)C)O)=O)CC2CCC(N(C)C(c3ccc(C(C)=O)cc3)=O)C2C1 63230,CCN1C(=O)Cc2cc(NC(N3CC(O)CC(C)(C)C3)=O)ccc21 63231,N1(C(c2nc(CC)sc2)C(=O)NCCCSC)CCc2nnnn2CC1 63232,C1(C(=O)NC2(c3ncc[nH]3)CC2)CN(C(C2CC(F)(CF)C2)=O)CC1F 63233,C(=O)(C1COc2ccccc21)N1CCC2(CC(NC(=O)C=CC3CCCO3)C2)C1 63234,C(=O)(C(F)C(C)CC(C)(C)C)N(CCC)CCNC(=O)C(C1CCCCCC1)O 63235,Cc1ccc(-c2nc(NC(N3CCN(CCN4CCCCC4)CC3)=O)cs2)cc1 63236,C(CNC(=O)CC1CC(F)(F)C1)(CC(=O)N(C)C(c1nccs1)C)OC 63237,c1(C(N2CC(O)(C(C(=O)NCCOCCCC#C)F)C2)=O)cnc(S)nc1 63238,CC1CS(=O)CCN1C(=O)C(Cc1cnc[nH]1)NC(C1CCC(C)(O)CC1)=O 63239,N1(C(C(C)C)=O)CCCC1(C)CNC(=O)Cc1cncs1 63240,C1(C(=O)NC(CN(C(c2sc(CO)nc2C)=O)CC)C)CCC2(CCOCC2)O1 63241,C1(NC(C2(CF)CC2)=O)CC2CC(NC(C3CC(O)C3)=O)CC12 63242,Cc1nccc(C(=O)NC(Cc2cn[nH]c2)C(=O)NCCCOC(C)C)c1C 63243,c1(CCNC(CCC=C(C)C)c2nnnn2C)c[nH]c2cccc(OC3CC3)c12 63244,Cc1nc2ccccc2cc1C(=O)N(C)CC1(NC(=O)C(O)CC[S+](C)C)CC1 63245,CC1(C(=O)O)CC(F)(F)CN1C(c1nc(C2CC2)n(-c2ccccc2)n1)=O 63246,C1(CC(N2CC(OCC(=O)NC)C2)=O)CCCCN1C(=O)C(F)SC 63247,C(=O)(C1CCCn2cc(C(C)(C)C)nc21)N(CCN(C)C(C1CC(Cl)(Cl)C1)=O)C 63248,Cc1cc(C2(c3noc(-c4sc(C)cc4Br)n3)CC2)n(C)n1 63249,C12CC(C13CCOCC3)N2.N1(CC)CC2CCCC(C1)N2Cc1ccccc1 63250,CC1CCC(C(N2CC(S(C)(=N)=O)C2)=O)CN1C(c1ccc(C(N)=O)o1)=O 63251,c1(C(N2CC3C(NC(c4ccc(I)cc4Br)=O)C3C2)=O)ccc2nc(O)oc2c1 63252,C1(C(=O)NC2C=C(C)CCC2)C(C)OCCN1C(=O)Cc1cccnc1C 63253,c1(C(=O)NC(C(C(C)C)NC(CCCC#C)=O)C)ccc2c(c1)CC2 63254,c1(C(=O)NC(CCCNC(C(C)OC)=O)c2ccccc2)cc(Cl)ccc1F 63255,N1(C(C2CCC(CNC(COC)=O)C2)=O)CC2OC(=O)N(C)C2C1 63256,C1(NC(CC=C=C)=O)CCN(C(=O)CN2CCCC2C)C12CC2 63257,C1(NC(C(CC)F)=O)CC(F)CN(C(c2ccccc2SC)=O)C1 63258,CC(C)CC(O)C(=O)N(C(C)C(=O)NCc1ncn(C(C)C)n1)C 63259,c1(CC)n[nH]c(CC)c1CC(=O)NC1CN(C(=O)COC2CC2)CC1C(F)(F)F 63260,C1(C(C)NC(c2cnn(CC3CCCC3)c2)=O)CN(c2cnc(F)cn2)CCO1 63261,N1(C(c2c(C)con2)=O)CC(CNC(=O)C=CCCc2ccccc2)CCC1C 63262,C1(C(=O)NC(C)CNC(C2(CF)CC2)=O)CCC2(CCC2)CC1 63263,c1(CCNC(c2[nH]c(=NCc3ccc(OC)cc3)sc2)=O)cccc(OCC)c1 63264,N1(C(CC(C)(C)OC)=O)Cc2nccn2CC(NC(C2(F)CCCCC2)=O)C1 63265,O=C1CC(C(=O)N2CCOCC(CNC(c3c(Cl)cncc3Cl)=O)C2)=NN1 63266,c1(C(=O)NCCC2(C(=O)NC3(CC)CCOC3)CCC2)ccnc(C)n1 63267,N1(C(=O)CC2CC3CCC2C3)CC2CCC1CN2C(c1cccc(C2CC2)n1)=O 63268,CC1=C(C(=O)NCCNC2CCC(Cl)CC2)SCCO1 63269,Cn1c(-n2nc(C3CC=CCC3)nc2CC(F)(F)C(C)(C)O)nc2ccccc12 63270,c1(CC(=O)NC2(COC)CN(C(c3sc(N(C)C)nc3C)=O)C2)ccc(Cl)nc1 63271,C(=O)(CCCCC(F)F)N(CC(CO)(CO)NC(C1C(C2CC2)C1(F)F)=O)C 63272,C1(NC(C(c2ccc(C)s2)C)=O)C=CCN(C(=O)Cc2cnnn2C)C1 63273,C(C)(CNC(=O)C=C(Cl)Cl)(C(C)C)NC(CCc1cc(C)[nH]n1)=O 63274,CC1(C)C(NC(C2CCC=CCC2)=O)CCN1C(=O)C(c1cc(F)ccc1F)=O 63275,c1(CCC(=O)N(C2CCCN(C(=O)CCC#N)C2)CC)cncnc1O 63276,c1(C(N2CCC(C(C)NC(=O)CC3(O)CCC3)C2)=O)ncc(F)cc1N 63277,c1(C(N2CCC(COC)(NC(C3CC(=O)N(C)C3)=O)C2)=O)c(Cl)ccnc1C 63278,C1(C(=O)NC(C2OCCN(C(c3c(OC)cncn3)=O)C2)C)CC2(CCOC2)C1 63279,c1(C(N(CCC)CCNC(C2CCC(C)S2)=O)=O)nc(C(C)C)ncc1NC 63280,N1(C(c2c(C(=O)OCC)c[nH]c2)=O)CCC(C)C(CNC(=O)CSC(F)F)C1 63281,c1(OC)cc(C(=O)NCC2CCN2C(C2CC(CF)C2)=O)cc([N+](=O)[O-])c1Cl 63282,Cc1c(N)ccc(C(=O)NCC(C)CNC(=O)CN2OC(C)(C)CC2=O)c1C 63283,c1(C(C)C)nc(NCC2CC2c2ccccc2C)cc(=NC(C)C2CCCC2)[nH]1 63284,N1(C(C(c2cscn2)OC)=O)CC(c2ccccc2)CC1C 63285,c1(C(N2CCC(CCNC(c3c(CCC)occ3)=O)C2)=O)cccc(F)c1Br 63286,CCC(C)(C(=O)N1CCC(OC)CC1)OCC1CCN(C(=O)C(C)(F)F)C1 63287,C1(NC(C=CCOC)=O)CC2CC1N(C(=O)C(F)C(C)(C)O)C2 63288,N(C1CN(C(c2nccn2CC)=O)CCc2ccccc21)C(C1(C=C)CCC1)=O 63289,C#CC(C)(C)C(=O)NC(CNC(=O)CCCn1cc(C)cn1)C(C)C 63290,c1(OC)cc2cc(C(=O)Oc3ncnc(-c4ccccc4)n3)[nH]c2cc1OC 63291,C(CC(F)F)(C(=O)NC1CCCN(CCO)C1)N(C(c1cn(CC=C)nn1)=O)C 63292,N1(CCC)CC(C(N2CCOC(CC(=O)Nc3cnn(CCF)c3)C2)=O)CC1=O 63293,C(CC(F)(F)C(=O)NC1CCC(=O)NC1)n1cc(CC(C)O)nn1 63294,N1(C(CC2C(C)(C)OCC2)=O)CC2(CCCC2)C1C(=O)NC1CN(C2CCC2)C1 63295,n1(CC)ncn(NC(=O)C(F)C(C)CNC(=O)CCc2ccc(C)o2)c1=O 63296,c1(C(=O)OC)ncccc1CN1CCC(F)(C(=O)Nc2ccc(SC)nc2)C1 63297,c1(OCC)ccc(Br)c(C(=O)NC(c2nn[nH]n2)C2CC2)c1 63298,CCCC(C)(CC)C(=O)N1CC(C(=O)O)C(CC(C)(C)C)C1 63299,C1(NC(C=C(C)Cl)=O)CC2CCC1N2C(c1c(C)nn(C)c1-n1cc(C)cn1)=O 63300,C(CC(C(=O)N1CCCCC1CNC(c1cc(C(C)=O)cs1)=O)N(C)C)SC 63301,N1(C(c2cc(OC)ncc2Cl)=O)CC2CN(C(c3ccc(C#N)o3)=O)CC2C1 63302,N1(C(c2c(C)scn2)=O)CCC2(C1)CN(C(c1nc(C3CC3)cs1)=O)CC(C)O2 63303,C#Cc1ccc(C(=O)N(C(C)C(N2CCCC(F)CC2)=O)CCC)cc1C 63304,CN(C)S(=O)(=O)NCC(=O)NC1CN(C(=O)C(=O)NC2CC2)CC1C(F)(F)F 63305,CN1CCC(C(=O)NCC2CC2NC(c2cc(C#N)c[nH]2)=O)CC1 63306,N1(C(C2CCSCC2)=O)CC2CCN(C(C3CCN4CCCC4C3)=O)C2C1 63307,N1(C(CC(=O)NCC#C)=O)CCC(NC(=O)C(=O)NCC)CC1 63308,Cc1cccc2[nH]cc(CN3CCCC(C(=O)Nc4ccc(O)c(F)c4F)C3)c12 63309,CCCCCC(CC)C(=O)N1CC(NC(=O)CC(F)(F)F)C(C)(C)C1 63310,C1(C(=O)NCC2CC(OC)C2(C)C)(CC)CCCN(C(=O)C(F)C(C)C)C1 63311,C1(CNC(C2(CCS(N)(=O)=O)CCC2)=O)CC2CC2N1C(=O)COCC1CCC1 63312,C1(NC(C(C)OCC=C)=O)C2CC1N(C(C1CCCCC1c1nc[nH]n1)=O)C2 63313,c1(C(N2CC(CC(=O)NC3CC34CCCC4)C3(C2)CC3)=O)cc2ncccc2[nH]1 63314,CN(CCc1ncc[nH]1)N1CCCC(CC2(C(N3CCOCC3)=O)CC2)C1 63315,CN1CC(C)(C)CC1C(N1CCC1CC(N1CCCC(CCF)C1)=O)=O 63316,c1(CNC(C2CC3CCC2N3C(C2C3CCCC23)=O)=O)cc(F)ccc1O 63317,CCCCCS(=O)(=O)CC(=O)N(CCC(C(C)(C)C)NC(=O)C(C)CSC)C 63318,c1(NC(C(CC#C)NC(c2cc(Cl)n[nH]2)=O)=O)ccc2c(c1)CCO2 63319,c1(C(=O)NC2C(SC)CN(C(=O)CCCc3ncco3)C2)c(C)nc(C)n1O 63320,N1(C(=O)CCCn2ccnc2)CC2CC(C1)N(C(=O)Cc1n[nH]cc1C1CC1)C2 63321,c1(C(=O)NC(CNC(c2c(C)nsc2NC2CC2)=O)C)nc2c(s1)COCC2 63322,Cn1c(C(N2CC(NC(c3ccc(C(C)(F)F)cn3)=O)C2)=O)cnc1S 63323,N1(C(C(CN(C)C)(C)C)=O)C2CCCC1CC(NC(c1cc(N)c(F)cn1)=O)C2 63324,C(=O)(C(=O)NOCCOC(c1ccc(F)cc1)Sc1cccc(Br)c1)OC(C)(C)C 63325,C(=O)(CCCCCCn1cc(C(O)C2CC2)nn1)N(CC(C)C#N)C 63326,CC(C)CC(CC(=O)NCCCCNC(=O)CC(C)C1CC1)CC(N)=O 63327,c1(C(N2CC(CNC(C34CC(C(F)F)(C3)C4)=O)C2)=O)cc2c(s1)CCCCC2 63328,C(C)(C(=O)N(C)OC)NC(c1cccc(OCCO)c1)c1n(CCOC)nnn1 63329,N1(C(c2ccc(NC(C)=O)s2)=O)CCC2CN(C(C3OCCC3C)=O)CC2C1 63330,O(NC(=O)C(c1ccoc1)NC(=O)CC1CC2CC2C1)CCCOC 63331,N1(C(NC2CNC(=O)c3c2cccc3F)=O)CCCC2(CCc3ccccc3O2)C1 63332,c1(C(N2CCC(CNC(C(C)CN(C)C)=O)C2)=O)n[nH]c2c1CCC2 63333,N1(C(C2CCC3N(C(c4c(C)ccnn4)=O)C2CC3)=O)CCc2ccncc2C1 63334,c1(C(=O)OCC)nn(C)c(C)c1COC(C1NC(=O)CC1C)=O 63335,C1(C(=O)NC(C#C)CCC)CC(C)CCN1C(C1CCC(OC)CC1)=O 63336,N1(C(c2c(C(C)=O)cn(C)n2)=O)CC(CNC(=O)C(C)O)OC2(CCC2)C1 63337,C1(NC(C(C)Cc2ccccn2)=O)COCCN(C(=O)Cc2cnnn2C)C1 63338,C1(NC(C2CC(OC)C2)=O)(CO)CCN(C(c2cn(C(C)C)nc2Br)=O)C1 63339,Cc1[nH]nc(C(F)F)c1C(=O)N(CC(O)CN(C)C(C1CCS1(=O)=O)=O)C 63340,Cc1ccc(F)cc1C(N1CC(CNC(=O)Cc2cn(C)nc2C)CCC1C)=O 63341,N1(C(C(C)O)=O)CCN2CCOCC2(CNC(C2CCS(=O)(=O)CC2)=O)C1 63342,Cn1ncc([N+](=O)[O-])c1C(=O)NC1C2CN(C(=O)COC(C)(C)C)CC12 63343,N1(C(C(C)(C)CNC(C2CC23CCOCC3)=O)=O)CC2CCCC(O)C2C1 63344,N1(C(=O)NC)CCCC2(NC(=O)CCOCC)CC2C1.N12CCC(CC1)C2=O 63345,C1(N(C)C(c2csc(Br)c2)=O)CCCC(O)C1 63346,N1(C(C2C(CCOC)C2)=O)CCC2(CCC(CNC(=O)COCC(F)F)O2)CC1 63347,C12(C(=O)NC3CCN(C(=O)CCC=CBr)CC3)CCCC1CCC2 63348,CCCCCCC(C)(F)C(=O)N1CCN(Cc2nc(-c3ccncc3)no2)CC1 63349,N1(C(=O)CC2CC23CC3)CC(C2CCCN(C(C3(F)CC4(CCC4)C3)=O)C2)C1 63350,C1(CNC(CCC=C)=O)CN(C(c2ccc(C(=O)C3CC3)cc2)=O)CC(C)(C)O1 63351,c1(C(N2C3CC(NC(C4CC(OCC)C4)=O)(C3)C2)=O)c(F)ccc(F)c1Cl 63352,Cc1ccc2c(c1)CC(C(=O)NCC(O)CNC(C1(C(F)F)CCC1)=O)O2 63353,C1(OCCOC)CC2CN(C(=O)C(c3ccco3)NC(=O)Cc3ccns3)CC12 63354,c1(OC)ccc(O)c(C(N2CCOC(CNC(=O)C(O)CC(N)=O)C2)=O)c1 63355,C(CN=c1cc(C)nc(-c2ccccn2)[nH]1)C1CN(C(C2C(C)(CC)C2)=O)C1 63356,c1(CC(N2CC(NC(Cn3c(C)ncc3)=O)C(C)(C)C2)=O)c[nH]c2ncccc12 63357,C1(C(N(C2CCCC(O)C2)C)=O)(NC(c2ccncc2N)=O)CCOCC1 63358,c1(CNC(CCOCC)C)cc(NC)cc(C(F)(F)F)c1 63359,N(C1CCOc2c(Cl)cc(Cl)cc21)C(C(N1CCCN(C(C)(C)C)CC1)=O)=O 63360,N1(C(C(CNC(CCC(=O)NCCC)=O)(C)C)=O)CCC(CO)C(C)(C)C1 63361,C1(C)(NC(C=C(C)CNC(=O)Cn2cnnn2)=O)CC2(CCC2)C1 63362,C(C(CC)(CC)C(=O)N1CC2CC(C)(C)C2C1)NC(C(CCC)OC)=O 63363,c1(C(=O)NC2C(C)CN(C(c3scnc3C3CC3)=O)CC2)ccc(S(N)(=O)=O)[nH]1 63364,Cc1oc(Cl)nc1C(=O)NC1(C(=O)N(C)Cc2cnn(C)c2)CCSC1 63365,c1(C(=O)NCCN(C)C(C2CCOC2=O)=O)ccc2c(c1)CNC2=O 63366,N1(C(Cn2c(C)ccn2)=O)CCC(C(N2CC(N3CCCC3)C2)=O)C1C(C)C 63367,N1(C(COC2(C)CCC2)=O)CC2COCC2(C(=O)NC(C(N)=O)C2CCCC2)C1 63368,N1(C(c2c(CC)[nH]nc2Cl)=O)CCCC2C1CCCN2C(=O)CSc1nc[nH]n1 63369,N1(C(c2ccc(NC)c(F)c2)=O)CC2CCC1CN2C(=O)CC(C)COC 63370,c1(CC(=O)NCCC2CCC(NC(CSC)=O)C2)ccccc1[N+](=O)[O-] 63371,c1(C(=O)NC(C2CN(C(C3(C#N)CCCO3)=O)C2)C)cc2nccnc2cc1F 63372,c1(CCC(N2C(CNC(C3CC3C(F)(F)F)=O)CC2)=O)ccc2c(c1)OCO2 63373,C1(c2ccccc2)(N(C)C)CCN(C(=O)CC2(C(c3ccccc3)=O)CC2)C1 63374,c1(CC(N2CC(CNC(C3C(=C)C3)=O)C(C)(C)C2)=O)nc2ncccn2n1 63375,c1(C(=O)NC(C)CCNC(C23CC(CO)(C2)C3)=O)cccc2[nH]ccc12 63376,C(=O)(C1=C(Cl)CCOC1)N1C(CNC(Cc2cncc(C#N)c2)=O)CCC1 63377,c1(NCC2N(CC)CCC2)nc(=NC2CC2CF)[nH]c2c(C)nn(C)c12 63378,c1(C(=O)NC2(CNC(C(=Cc3cccs3)C)=O)CC2)cc2ccc(Cl)c(F)c2[nH]1 63379,c1(C(N(CC2C(C)CCC2)CC2CC2)=O)ccc(N2CCOCC2)cc1Cl 63380,C(C(CC(C)C)C(=O)N1CCC(NC(c2nc3ncccn3n2)=O)C1(C)C)OC 63381,N1(C(c2n(CCC)ncc2)=O)CC2CC1C2NC(c1ncccc1OC)=O 63382,C1(CNC(C=CCCC)=O)CC(OC)CN1C(c1cnc(O)o1)=O 63383,c1(OC)cnc(F)c(C(=O)NC(C)CNC(c2nc(=O)n(C)[nH]2)=O)c1 63384,N1(CC(C)C)CCC(C(N2CCC(NC(=O)CC3CN(C)CC3O)C2)=O)CC1 63385,Cc1cnc(NCc2cc(C)no2)c(S(=O)(=O)NCC2(CO)CC(C)C2)c1 63386,CCCC(C)(O)C(=O)N1CC(CCNC(=O)C(c2ccccc2F)C)(OC)C1 63387,C#Cc1cc(C(=O)NC2CCC(NC(=O)C(C)O)CC2)cc(N)c1 63388,c1(C(=O)NC2CN(C(C3N(C)CCOC3)=O)CC2(C)C)c(Cl)nc2ccccn12 63389,C1(CC)CCN(C(=O)Cc2ccccc2C)C1C(=O)NC1CCCC1C#N 63390,c1(CN2C(CC(=O)NC3(C#N)CCOCC3)CCC2)c[nH]c2nc(Cl)ccc12 63391,C(C(C(=O)NCc1cc(OC)ns1)C(C)(C)C)NC(CCOCC)=O 63392,Cc1cccc2[nH]c(=NCCN(C(=O)CC3CC3C)C)oc12 63393,N1(C(CCOCCCC)=O)CCC(NC(=O)C(CC)N(C)C)C(CO)CC1 63394,Cc1ccc(NC(N2CC=CC2C(=O)NCC2(Br)CC2)=O)cc1 63395,c1(C(C)NC(CC2N(C(CC=C)=O)CCOC2)=O)cc(F)c(Cl)cc1Cl 63396,c1(C(=O)NC2CC(NC(C3N(C)CCC3)=O)C2)c2c(nn1C)CCC2 63397,C1(C(=O)NC(c2nc(CC)on2)C)CCCCCCN1C(=O)CC(C)O 63398,C(=O)(C(F)CCC(C)C)N1CC(NC(c2[nH]cc(C)c2)=O)C(O)C1 63399,c1(C(=O)OC)ccc(N2CC(CNC(=O)NC(C)CN(C)C)C2)nc1 63400,N1(C(c2c(C)n[nH]c2)=O)CCCC(C(C)NC(=O)Cc2csc(S)n2)C1 63401,C(=O)(C1CCOc2ccccc21)NC(C)CN(C)C(c1c(Br)cnn1C)=O 63402,N1(C(C(CC)SC)=O)CCOCC(NC(=O)C(C)OC2CCOC2)C1 63403,CCC(C)C(O)CNC(c1ccc(OC2CC2)cc1)c1ccn(C)n1 63404,N1(C(CC(C(F)F)NC(C2CCCC23CCC3)=O)=O)CCCC2CNC(=O)C12 63405,C1(O)(CCNC(C2(CC#C)CCCC2)=O)CCN(C(c2ccnn2C(C)C)=O)C1 63406,C1(C#N)(C(N(CCC(C)NC(C(C)N2CCC2)=O)C)=O)CCSCC1 63407,N1(C(C2N(C(c3c(C)c[nH]n3)=O)CCCC2)=O)CCOCC2(CC2)C1 63408,Cc1cn2nc(C(=O)N(CC(C)(C)CNC(=O)CC3CSC3)C)cc(C)c2n1 63409,C1(C(C(=O)NC(CCOC)CNC(c2cnccn2)=O)C)CCN(C(C)C)CC1 63410,Cn1cnc(NC2CCC(NC(=O)CCc3ccncc3)CC2)cc1=O 63411,C1(CNC(C(CCC)OC)=O)CCN(Cc2nnc(Cn3cccn3)o2)CC1C 63412,N1(C(C)=O)CCCCC1C(N1CCC(CNC(=O)CCCc2csc(C)n2)C1)=O 63413,C(C1CCOC1)=CC(=O)NCCC(O)CNC(=O)C(F)(F)C1CCCC1 63414,CC(C)(CCCC(=O)NCC1CCCC1O)NC(=O)C(N)=O 63415,C(=O)(C(CC)CC=CC)N1CCCC(CCC(=O)NCC(=C)CC)C1 63416,C(CN=C(NCc1ccnc(N2CCOC(C)C2)c1)N(C)CC(C)C#N)OC 63417,C1(CNC(C2CC(NC(C(COCC)C)=O)C(O)C2)=O)NC(=O)CC1(C)C 63418,c1(C(c2nnnn2CC(F)F)NCc2cn(C)nc2Cl)cc(S(C)(=O)=O)cs1 63419,CC1OC2(C(=O)NCC3CCN(C(=O)CN4CCN(C)CC4)CC3)CCC1C2 63420,CCC1=C(C(=O)N2CC3CC2CCC3NC(c2ccnc(F)c2)=O)CCCO1 63421,C1(C2CCC2)(C(=O)NC(CC)CNC(=O)CC(C)(C)SC)CC1(F)F 63422,C1(C(=O)NC(CC)(CNC(=O)COC)CC)C2Cc3c(Br)cccc3C12 63423,c1(SCC(=O)NCC(CC)NC(c2cccs2)=O)ccccc1N=NN(C)C 63424,n1(CC)c(CNC(=O)CC(C)(C)NC(=O)C(C)=C2CC2)nnc1O 63425,C1(CNC(C2CC3C=CC2C3)=O)CN(C(c2cocn2)=O)CCC12CCOCC2 63426,C12(C(=O)NC3CN(C(Cn4c(C)ccn4)=O)CC3C(F)F)CC1COC2(C)C 63427,c1(C(N2CC3CC2CN3C(c2cc(F)ccc2F)=O)=O)cccc(F)c1O 63428,c1(C(=O)NC2CC(NC(c3ccccc3-n3ccnc3)=O)C2)cc(F)ccc1Cl 63429,c1(CCC(=O)N(CCC(C)NC(=O)C#CC2CCC2)CC)cc(F)c(F)c(F)c1 63430,Cc1cccc(C(N2CC3(NC(c4ccsn4)=O)CCC2C3)=O)c1Cl 63431,c1(CC(=O)NCC(C)NC(C2C(C(=O)OC)CC2)=O)coc2c(C)c(C)ccc12 63432,c1(C(=O)NCC2(NC(=O)CN3CCCC3=O)CCC2)cccc2cccc(O)c12 63433,N1(C(CN(C(COC)=O)C)=O)CC(NC(=O)C(C)(C)C2CCC2)C(O)C1 63434,N1(C(C(C)NC(CC)(C)C)=O)CCCC1(C(=O)NC(CO)C(C)C)CC 63435,N(C(=NCc1ccc(C(N)=O)cc1)NS(=O)(=O)CC1CCCO1)C1C(C)(C)CC1 63436,C(CC(C)(C)C)(C(=O)N1CC(O)C(C2CC2)C1)NC(C(CC=C)OC)=O 63437,c1(OCC)nc(N2CC(NC(c3ccno3)=O)C(O)C2)ncc1OC 63438,C(=O)(C1=CCC(F)(F)CC1)N1CCC(CCNC(CCC(C)OC)=O)C(F)(F)C1 63439,N1(C(CC(CC)C)=O)C(CC(=O)NC2CCCCCC2C)C2CCCC12 63440,C1(CC)CCN(C(=O)CCc2cn(C)cn2)C1C(=O)NCC#CCOC 63441,C(=O)(CCC(C)CN(C)C)NCC1(F)CN(C(C(C)NC(C)=O)=O)C1 63442,C1(C(CNC(CCC)=O)Cc2ccccc2)CCN(C(c2ccoc2Cl)=O)CC1 63443,c1(CN2C(c3cccc(OC)c3)CC2)cccc(C)c1OC1CCOC1C 63444,C=CC(CC)C(=O)N1C(C(N2CC(C)(CO)C2)=O)CC1C 63445,N1(C(CC=CCC)=O)CC2(CC(NC(C3(CC)CCC(=O)N3)=O)C2)C1 63446,CC1=C(C(=O)NCC2CCCN2C(c2cnn(C)c2)=O)CCC1 63447,N1(C(CCC2CCCN(C)C2)=O)CCN(C)CC1CNC(=O)CCNC(=O)CO 63448,Cc1cc(CNC(C2COC(CNC(c3sccc3C)=O)C2)=O)cc(C)c1 63449,c1(C2(C(=O)NCC3N(C(C(COCC)C)=O)CCC3)CC2)ccccc1F 63450,Cc1cccc(CC(=O)NC2CC(O)(CNC(=O)C(O)C(C)(C)C)C2)c1C 63451,N1(C(C(CCC2CC2)NC(c2c(OC)ccs2)=O)=O)CC2COC(=O)C2C1 63452,C1(CCNC(C2(C)CCCC2)=O)CC(F)(F)CN1C(c1cc(CO)ccc1Cl)=O 63453,C1(NC(C(=O)NCCOC)=O)CCC(C)N(C(c2ccc(N)cc2F)=O)C1 63454,c1(-c2cn(CC(N3CC(C)C3C(N3CCCC3)=O)=O)nn2)ccc2ccn(C)c2c1 63455,c1(CC)ccc(C)c(C(N2CCC(NC(=O)C(c3cccnc3)O)C2)=O)c1 63456,CC(CCCC(=O)NC(C)(C)CC1CCOC1)NC(c1cc(Cl)no1)=O 63457,c1(C(=O)NCCC2CN(C(=O)CCC3CC3(Cl)Cl)C2)ccc[n+]([O-])c1 63458,C1(C(=O)NCC(=C)Cl)CC2CC1CC2NC(=O)CC1CNC(=O)O1 63459,Cc1nc(C(=O)NC2CN(C(C3CCC3c3nc[nH]n3)=O)C2)cn(C)c1=O 63460,c1(C(=O)NC2CN(C(COC)=O)CC2C)cc(C(F)(F)F)c(OC)c(C(F)F)c1 63461,c1(CC(=O)NCC(CNC(C2CC(C(F)F)C2)=O)OC)ccc2c(c1)OCCO2 63462,c1(CNC(c2ccc(CC)o2)=O)c(C)nn2c1CN(C(C1(C)CC1F)=O)CC2 63463,N1(Cc2c3cccc(C)c3[nH]c2)CCc2ncc(Br)cc2C1 63464,c1(C(=O)NC(CNC(C(C(C)C)N(CC)CC)=O)CC(C)C)ccc(N)c(Cl)n1 63465,C=CCC(F)(F)C(=O)NCC1CC(C)N(C(=O)C#CC2CC2)C1 63466,O=S(=O)(CCO)CCNC(=S)NC1CCCCCCC1 63467,c1(C(N(C)CC2N(C(CCOCC)=O)CC(F)C2)=O)cc2n(n1)CCC2 63468,c1(C(=O)NC2CN(C(c3c(C)ocn3)=O)CC3C2C3)ccnc2ncccc12 63469,c1(OCC(N2C(CNC(=O)CCCF)CCC(C)C2)=O)cccc(S(C)(=O)=O)c1 63470,c1(C(N2CCN(C)C(CNC(=O)CCOC3CC3)C2)=O)cccn2nnnc12 63471,C1(N(C(C(C)NS(CC)(=O)=O)=O)C)CCCCC1N(C)C(c1cccc(C)c1)=O 63472,N1(CC(C)NC(c2cc(C(C)=O)on2)=O)CCN(C(=O)Cn2nnc(C)n2)CC1 63473,C12(C(=O)NCC3N(C)CCN(C(CC(C(=C)C)O)=O)C3)C3CC(CC13)C2(F)F 63474,C(=O)(C(C)CC)N(CC(=O)N(CC(CSC)O)C)CC1CC1 63475,c1(N2C(CNC(C3(C)CCC(=O)N3)=O)CC(F)(F)C2)ccc(S(C)(=O)=O)cn1 63476,C1(C(=O)NC2CN(C(C(C)Oc3ccc(Cl)cc3)=O)C2)CC2(CCC2O)C1 63477,CN=c1cc(C(N2CCCC(CO)(NC(c3cc(Br)oc3C)=O)C2)=O)cc[nH]1 63478,c1(C(=O)NC2C(NC(c3cn(CCO)nn3)=O)CC2)cccc2cnsc12 63479,CC(CC(=O)N1CCC(NC(c2cc3n(n2)CCOC3)=O)C1)CC(F)(F)F 63480,c1(NCCCCSC)ncccc1S(=O)(=O)NC1COC2(CCC2)C1 63481,C(C(C)(C)C(=O)NCC[Si](C)(C)C)N(C)C(c1ccc(C2CC2)o1)=O 63482,c1(C(N2CC(N(C(C(CC)C#N)=O)C)C3(C2)CC3)=O)c(F)cc(OC)c(F)c1F 63483,C1(C(=O)NC2CN(C(c3c(CCC)nsc3N)=O)C2)CC2(CCCC2)CO1 63484,C1(NC(=O)CCc2ccccc2)CN(Cc2cccnc2F)CC(F)(F)C1 63485,C12(CNC(CN(CC)CC)=O)CC(NC(=O)CCc3cccnc3)(C1)C2 63486,N#Cc1ccnc(C(N2CCC(NC(C3CCCC(F)(F)C3)=O)CC2)=O)c1F 63487,C(=O)(CCCCC(F)(F)F)NCCCCn1cc(CNC(C)=O)nn1 63488,C=CC(C)(O)C(=O)N1CCC(CF)(NC(=O)C(C)(C)COC)C1 63489,C12(NC(Cc3n(C)ncc3)=O)CCN(C(c3cc4sccc4s3)=O)CC1C2 63490,N1(C(CCn2cnc(=N)[nH]2)=O)CCN(C(C23CCC(C2)C3)=O)CC1CCO 63491,Cc1cc(C)c2[nH]c(C(=O)NC3CC3NC(=O)CNS(=O)(=O)C3CC3)cc2c1 63492,c1(OCC)cc(NC(C)CCNC(=O)C(O)C2CC2)ccc1[N+](=O)[O-] 63493,Cc1cc(O)ncc1C(=O)NC1CC(O)CN(C(c2ccnc(C(C)C)n2)=O)C1 63494,N1(C(C(CNC(C2CC3(CC(C)C3)C2)=O)(C)C)=O)CCN(C)C(C)C1C 63495,Cc1csc(C(=O)NCCCNC(c2c(C3CCCCC3)noc2C(C)C)=O)c1C 63496,C1(CNC(C(C)OCC)=O)C2CCCC1N(C(c1ccnc(C(N)=O)c1)=O)C2 63497,C1(CC(N2CCC(C)(N(C)CC)C2)=O)C2CCCC2N1C(C1CC12CC2)=O 63498,c1(N2CC3C(NC(C(CC)C4CCOCC4)=O)C3C2)cc(S(C)(=O)=O)ncn1 63499,C(=O)(C(Cc1cnc[nH]1)N1CCCC1CN(CC(=O)OC(C)(C)C)C)NC 63500,O=C(CCCCCNC(=O)CC1CCSCC1)NOCCc1ccncc1 63501,C1(C)(NC(C(CCC)O)=O)CCC(NC(c2ccc(CO)c(Cl)c2)=O)CC1 63502,CN1CCC(C2(C(=O)NCC(F)CNC(c3c(F)ccc(O)c3F)=O)CC2)CC1 63503,NS(=O)(=O)c1cccc(C(=O)NC2CC(CNC(C3CC3(Cl)Cl)=O)C2)c1 63504,N1(C(Cc2cc(C)sc2)=O)CC(CNC(=O)CCOC2CCC2)C2(CC2)C1 63505,N1(C(C(C)SCCCC)=O)CCC(NC(c2cc(C(C)=O)cs2)=O)C(C)C1 63506,C1(CN(C(C(CC=C)N(C)C)=O)C)CCCN(C(C2CCCCCC2)=O)CC1 63507,c1(CC=CCC(=O)N(CC(C)NC(c2nn[nH]c2Cl)=O)C)ccccc1 63508,C(=O)(C(C(C)C)C(C)C)N1CCOCC(C(=O)NCC(COCC)O)C1 63509,C(=O)(C1CCc2nccn21)N1CCCC(O)(CNC(C2N(C)CC3(CC3)C2)=O)C1 63510,CCC(CC(C)C)C(=O)N(C(C)C(=O)NCC(CC)OC)C1CC1 63511,c1(C(=O)NCC2N(C(C(CCC)(C)C)=O)CCCC2)cc2n(n1)CC(C)NC2=O 63512,c1(C(N2CC(N(C(C3C(C(C)C)C3)=O)C)C2)=O)cc(N)cc2ccccc12 63513,c1(C(=O)OC)ccc(C)nc1N1CCCCC(NC(=O)CCCCN(C)C)C1 63514,CC(CC(=O)NCCN(C(=O)Cc1ccccc1)C1CC1)n1ccnc1 63515,C12(C(N(C(C)C(F)F)C)=O)CC(n3cc(CNC(N)=O)nn3)C1C2 63516,Cc1nc(C(=O)NCCC2(NC(=O)CN(C3CCC3)C)CC2)n[nH]1 63517,Cc1c(-n2cc(CNC(C3(NC(c4ncccc4O)=O)CC3)=O)nn2)cnn1C 63518,C1(C(=O)NC2CC(CCNC(c3c(CC)ocn3)=O)C2)CCCC(C)(C)O1 63519,CCC(F)(F)CC(=O)NCc1ncoc1CCNC(=O)C(C)(O)CCC 63520,C1(CNC(C2C(CC)C2)=O)CN(C(c2cc(F)ccc2C(F)F)=O)CC1(F)F 63521,c1(OC)cc2nc(O)n(CN3C(C)CCC3C)c(=O)c2cc1OC 63522,Cc1ccc(C(=O)NCC(C)NC(=O)C(c2c(C)n[nH]c2C)C)c(N)c1Br 63523,C1(NC(C2(CC)CCCN2C(=O)C(F)C2CCCC2)=O)CCC2CC1CO2 63524,Cc1cc(C(=O)N(CC(O)CN(C(=O)CC(C)F)C)C)nn1-c1ccc(Cl)cc1 63525,C1(C)(NC(CCCn2cc(CNC(CCC(=O)OC)=O)nn2)=O)CCCCC1C 63526,c1(C(N2CC3CC(C2)N(C(C2COCCOC2)=O)C3)=O)c(F)ccc2c1OCC2 63527,C(CC)(CC(=O)N1CC(C)(C(N)=O)C1)NC(c1n(CC#C)ccc1)=O 63528,C1(NC(c2c(CC)cno2)=O)CC2CC1CN(C(c1ccsc1C)=O)C2 63529,CC(CC(=O)NCC1CC1NC(=O)CC(=O)NC1CC1)P(C)(C)=O 63530,Cc1ccc(OCCN2CC3C(NC(=O)C(C)CCN(C)C)C3C2)cc1 63531,C1(CNC(C(C2CCCO2)NC(C2CC=CC2)=O)=O)CC(C2CC2)=NO1 63532,c1(CC(N2C(CNC(C(CC#C)C)=O)CC3(CC3)C2)=O)cccc2c1CCC2 63533,C1(NC(=O)OC(C)(C)C)COC2(CCC2)CN1N1C2CCCC1C2 63534,CCCCCC(O)C(C)C(=O)N1CCCC(CCNC(C2CCN2CC)=O)CC1 63535,C(C1CCC(C)CC1)=CC(=O)N(C1CCCN(c2ccc(C#N)nc2)C1)CCC 63536,CC1(C(=O)NC(C)(CNC(=O)Cn2ccc(C3CC3)n2)C2CCC2)CCCCO1 63537,C1(CC(=O)NCC(C)CNC(=O)C(F)(F)c2csc(=N)[nH]2)CC(=O)NC1=O 63538,N1(C(c2c(C)csc2)=O)CCC(C)(C)C1C(=O)NCC1CCCCC1(C)C 63539,C1(C(=O)NCC2(F)CC(NC(CCNC(C)=O)=O)C2)CCCC(O)C1 63540,CC1CN(C(=O)CN2CCCCC2C)CC1NC(c1ccc(Cl)cc1)=O 63541,C1(C)(C(=O)NC(CNC(C(CCCC)O)=O)CCOC)CCCCCCC1 63542,c1(CN2CC(C(=O)Nc3ncc(F)cc3Br)C(O)CC2)ccc2ncnn2c1 63543,C(=O)(C(F)C(F)(F)F)NCCC1CC(NC(c2cc(C)n(C(C)C3CC3)n2)=O)C1 63544,CC1CC(C(=O)NCCC(=O)N2CC(N(CC(F)F)C)C2)CCS1 63545,c1(CCC(=O)OC)ccc(NC(C2CCCOC2)=O)c(C)n1 63546,C1(NC(CCc2cn(C)nn2)=O)CN(C(C2(O)CCOC2)=O)CC(C)(C)C1 63547,N1(C(CSCC(=O)OC)=O)CCN(C(=O)CCc2cncn2C)CC1C1CCC1 63548,C1(NC(C2CC(C)C2)=O)CC(C)CN(C(=O)NCCC(=O)OC(C)(C)C)C1 63549,N1(C(C=CC(CC)=CC)=O)CCC(C)(C)C(CNC(C2CCCC3(CC3)C2)=O)C1 63550,N1(C(C=CCC)=O)CC(CNC(=O)Cc2cnn(C(CC)CC)c2)CC1C 63551,CN1CCc2cc(C(=O)NC3COCC3NC(=O)C(O)CC(C)(C)C)ccc2C1 63552,C#CCCC(C(=O)NCCCC(O)CO)NC(=O)CCC=CCC=C 63553,C(CN=C(NC(c1cccs1)C1CC1)N1CC2CCOCC2C1)c1ccsc1 63554,N1(C(COCCCCC)=O)CC(C)(CNC(c2cc(SC)c(C)o2)=O)CC1(C)C 63555,c1(C(=O)NCC=CCNC(CCC(C)C#N)=O)cc2n(n1)CCCN2 63556,C(=O)(CC1=CCN(C)CC1)NC1CCN(C(C(C)C(F)(F)F)=O)C(C)C1 63557,C(N=c1[nH]c(Cl)nc2cccc([N+](=O)[O-])c12)C1(O)CN(C(C(C)C(C)(C)C)=O)C1 63558,Cc1cc(C(N2CC(NC(C3(CO)CCCO3)=O)C(O)C2)=O)cc(Cl)c1 63559,c1(CC)nc(NN(C)C(=O)OC)cc(=NCC(c2cccs2)N(C)C)[nH]1 63560,N1(C(CN(CCC)C)=O)CCC2(CCN(C(C3CCOC(C)C3)=O)C2)C1 63561,Cc1cc(=NCC2(C)CCC(C)(C)CC2)[nH]c(=NCCCC(C)O)[nH]1 63562,N1(C(=O)CN2CCN(CCO)CC2)CCN(C(C2(F)CC=CC2)=O)CC1C1CC1 63563,C1(C)(CC)CCC(C(N2CC(N(C)C(c3csnc3Cl)=O)C2)=O)O1 63564,C12(NC(C(CC(C)C)C)=O)CCCN(C(=O)COC3(C)CCCC3)CC1C2 63565,N1(C(COCC(N)=O)=O)CC(C2(NC(=O)Cn3ccc(O)nc3=O)CC2)C1 63566,O=C1NC(=O)N2CCN(C(=O)NC3CCC(C4CC4)CC3)CC12 63567,N1(C(CCO)=O)CCN(C(=O)CC2CCCC(C)C2)CC1.C(=O)OCC 63568,C12(C(=O)OCC)CC(CC(N3CC(O)(CNC(=O)C=CCO)C3)=O)(C1)C2 63569,N1(C(CCNC(C)=O)=O)CC(NC(c2c[nH]c(C(N)=O)c2)=O)CC(F)(F)C1 63570,C1(O)(C(=O)NC2CN(C(c3c(CC)noc3)=O)C(C)CC2)CCC(C)(C)CC1 63571,C1(C2(O)CN(C(C3CCc4nn[nH]c4C3)=O)C2)(CNC(CCNC(N)=O)=O)CC1 63572,c1(-c2cn(C(C(=O)N(C(COCC)C)C)C)nn2)[nH]nc(C(=O)OC)c1Br 63573,C#CCCCCCC(=O)N1CC(OC)C(NC(C2(C(C)C)CNC(=O)C2)=O)C1 63574,N1(C(COC(C)C)=O)CCCC(C)(C)C1C(=O)NC(CC1CCCC1)CO 63575,N1(C(C2(CNC(C(COCC)C)=O)CC=CC2)=O)CCCSCC1C 63576,c1(C(=O)OC)cnn2c1CC(NC(N1CCC(C)(C)CC(C)(C)C1)=O)CC2 63577,C1(N(CCC)C(C2CC2CF)=O)CCN(C(=O)C(F)(F)C2(OC)CCC2)C1 63578,C12(C(=O)NCC3(O)CCN(C(=O)Cc4cnc[nH]4)C3)CC3CC(CC1C3)C2 63579,c1(C(=O)O)nnc(CNC(=O)C(O)CC2CCOCC2)s1 63580,C1(C(F)(F)F)(NC(c2ccn(C)c2)C)CCCCCC1 63581,CC(CC(F)(F)F)C(=O)N(C1CN(C(C2CC(n3cnnc3)C2)=O)CCC1O)C 63582,Cc1csc(C(=O)NCC2CN(C(N)=O)CC2C)c1Br 63583,c1(-n2cc(C(=O)OC)nn2)cccc(NC(c2ccoc2)C)c1 63584,CCC(CC#N)N=c1ccc(Br)c(S(=O)(=O)NCCS(=O)(=O)NC(C)C)[nH]1 63585,C(C(=O)NCC(C)CN(C)C(c1c(NC(C)=O)c[nH]c1C)=O)(C(C)C)OC 63586,N1(C(Cc2ccc(OC)c(Cl)c2)=O)CCN(C(=O)C(C#N)C2CC2)CC(C)(F)C1 63587,N1(C(=O)C=Cc2ccco2)CCC2CCN(c3c(Cl)cncc3[N+](=O)[O-])CC2C1 63588,c1(C(N(C(CNC(C2(CCC=C)CCCC2)=O)C)C)=O)nccc(Cl)c1O 63589,c1(NC(C2C3(CC(NC(=O)OC(C)(C)C)C3)C2)=O)cc(Cl)c(F)cc1S(N)(=O)=O 63590,CCCCC(CC)C(=O)NCC1CCCN(C(=O)CC2CCOC(C)(C)C2)C1 63591,N1(CC(=O)NC2CCOCC2NC(C2CC(=C3CCC3)C2)=O)C(=O)CCC1=O 63592,Cc1cc(C(N2CCC(F)(C(N3CCC3C(C)O)=O)CC2)=O)nc(O)n1 63593,c1(CC(N2CCN(C(c3c(C)nn(C(C)C)c3)=O)CC2)=O)ccc(F)cc1F 63594,C(=O)(CC(C)(C)C(=O)NC1CCC(NC(=O)CC2CCC(C)(C)O2)C1)OC 63595,C1(NC(CCC(=C)Cl)=O)CN(C(=O)COc2cc(Cl)ccc2C)CC12CCC2 63596,CC1CC=CCC1C(N1CCN(C2CN(C(C3(O)COC3)=O)C2)CC1)=O 63597,C1(NC(=O)OC(C)(C)C)CN(C(=O)CCCCc2cnn[nH]2)NC1=O 63598,N1(C(CCC(C)OC)=O)CCCC2(NC(=O)C(N3C(C)CCC3C)C)CCCC12 63599,c1(C(=O)Nc2ccc(NC(C(CCC)CC)=O)cc2C)cnc2c(c1)NCC(=O)N2 63600,N1(C(CNS(NC)(=O)=O)=O)CCCN(C(C2CC(O)C2)=O)C(C(C)C)C1 63601,C1(C(=O)NC2(COC)CN(C(=O)CC3COCCN3C)C2)CCCCN(C)C1=O 63602,c1(C(N(CCCC)C)=O)ncsc1Br.c1(C(C2C(C(=O)OC)C2)=O)ccccc1 63603,Cc1nccc(N2CCC(C)(C(=O)NCc3cccc(C(F)(F)F)c3)C2)n1 63604,C1(C(=O)NC(C)CNC(=O)C(C)(C)n2cc(Cl)cn2)CCC(=O)NC1 63605,C1(C(=O)NCCCCC(=O)NC)CCC2(CC2)N1C(=O)C(c1cncn1C)O 63606,Cn1c(N2CCOC(CNC(=O)CC3CCC(F)(F)C3)C2)cc(=O)n(C)c1=O 63607,c1(OC)c(C(C(=O)NCCC#N)N(C2CCOC(C)C2)C)ccnc1F 63608,C=C(CC(C(=O)NCCNC(=O)OC(C)(C)C)N(C)C)c1ocnc1C 63609,c1(CN2C(C(=O)Nc3cc(C)c(Cl)cc3Cl)CC3CC32)ccc2c(c1)C(=O)CC2 63610,N1(Cc2scc(C(=O)NC(Cn3c(C(C)C)nnn3)=O)n2)CCC(N(C)C)CC1 63611,N1(C(Cc2nc(C)sc2C)=O)CCC2(CC1)CC2CNC(C1(C#N)CCOC1)=O 63612,N1(C(C=C=C(C)C)=O)CCN(C(=O)CC(C)n2cccc2)C(CC(F)F)C1 63613,C(=O)(C(CC(C)C)ONC(c1cnsc1C)=O)NCc1nc(COCC)sc1 63614,CC1CCN(C(C2(CO)CC(F)(F)C2)=O)CCN1C(=O)Cc1cnns1 63615,Cc1nccn1CCCC(=O)NC1CCC(CC(N2CCCC2C)=O)C1 63616,C(=O)(CC(C)(O)C(F)(F)F)N1CCCC(CNC(C2(SC)CC2)=O)CC1 63617,c1(NC(C(=O)NCC(C)NC(c2cccnc2Br)=O)=O)cccc(OC(F)F)c1 63618,C1(NC(C=Cc2n(C)ncc2)=O)CN(C(=O)Cc2n[nH]c(=N)s2)CC1S(C)(=O)=O 63619,c1(C(N2CC3C(NC(CCCC#C)=O)C3C2)=O)cc(C)nc(N(C)C)n1 63620,CC1(C)CN(C(=O)C(C2(O)CCC2)NC(C2CCC(=O)CC2)=O)CCC1CO 63621,C(=O)(CCC(C)(C)C)N(C(CCNC(C(CN(CC)CC)F)=O)C)C 63622,c1(C(=O)NC2CC(NC(c3ccn4c3CCCC4)=O)C2)cnn2c(=O)cc[nH]c12 63623,C1(C(N(C(CCNC(C)=O)C)C)=O)CC2CCC1O2 63624,C(=O)(C(F)CC(C)(C)N)NCCc1nnc(C(=O)OC)s1 63625,N1(C(C(C)(C)OC)=O)CCN(C(c2ccc(C#N)c(F)c2)=O)CC(C)C1 63626,C(=O)(C(C)(O)C(C)(C)C)NC1C(NC(c2ccc(CC)nc2C)=O)CCC1 63627,C12(NC(c3ccc(Cl)cc3F)=O)COCCC1CN(C(c1ccns1)=O)C2 63628,c1(C(=O)NC(C)CCN(C)C(C2CC2C)=O)cc(-c2ccncc2)nn1C 63629,c1ccc(N2CC(C(C3CCCCC3)NC3CCNC3)C2)cc1 63630,Cc1cncc(CCNC(=O)C(C2CCN(C(c3cnncc3O)=O)CC2)C)n1 63631,N1(C(C)(C)C)CCN(C(F)(F)F)C(=O)C1.c12cnc(nc1)CCNC(=O)C(=O)N2 63632,Cc1c(Cl)ccc(C(=O)NCC(C)(C)CNC(=O)C2=NNC(=O)CC2)c1N 63633,c1(OC)ccc(CC(C)C(=O)OC)cc1S(=O)(=O)NCCc1cc(C)n(C)n1 63634,C12(OC)CCC(CN(C3CCOC3)CCO)(CC1)C2 63635,c1(NC)ccc(C(N2CCCC(CCCCNC(=O)C3CC3)C2)=O)nc1 63636,c1(C(=O)NC2C(CNC(C3CCC(C)CC3)=O)CCC2)cccc2cncn12 63637,N1(C(Cc2c(C)scc2)=O)CCC(NC(=O)C=Cc2ccoc2)C(C)C1 63638,c1(OC)cc(C)c(C(=O)NCCN(C)C(c2nnn(C)c2C(F)F)=O)cc1Cl 63639,C(=O)(C(F)C(C)(F)F)NC(C(=O)NC(c1nc(CC)on1)C)(C)CSC.C(C)(=O)O 63640,c1(C(=O)NC2CC3CN(C(C4(NC(N)=O)CC4)=O)C2C3)c(Cl)cc(Cl)nc1N 63641,C(=O)(C(C)(C)CCCO)N(C)CC1CCCN1C(c1ccc(C(F)F)cc1)=O 63642,N1(C(N2CCN(C(C)=O)CC2)CC)C(=O)CCC1=O.C1(=O)CO1 63643,c1(C(N(CCC(C(C)C)NC(C(CC(=O)OC)C)=O)C)=O)cc2cn[nH]c2cn1 63644,O=C(C1CCCc2scnc21)NC1CCN(C(=O)CCOCC(F)(F)F)C12CC2 63645,C1(CC(=O)N(Cc2scc(C(=O)NCCc3c(C)ocn3)c2)CC)CCCNC1=O 63646,C1(N(C(=O)COCP(C)(C)=O)C)CN(C(C2CCN(CC(F)(F)F)C2)=O)CC12CC2 63647,C12(C(=O)NC3C(NC(COC(C)(C)C)=O)COC3)C3C4C1C1C2C3C41C(N)=O 63648,C1(NC(C2N(CC)CCOC2)=O)CCN(C(=O)Cc2cccs2)CC1C 63649,N1(C(C(CC)(C)O)=O)CCCCC(NC(c2ccsc2Br)=O)CC1 63650,Cc1c(C(N2CCCN(C(C3OCCO3)=O)C(C)C2)=O)[nH]c2cc(F)ccc12 63651,C(=O)(CCC(=O)N(C(C)(C)CNC(C1CCCC(F)C1)=O)CC)OCC 63652,C1(CNC(COCCCC#C)=O)CC(C)CN(C(c2occc2CC)=O)C1 63653,C1(NC(c2n(C)ccn2)=O)CN(C(C2CC2C(C)(F)F)=O)C(C)(C)C1 63654,c1(C(=O)NCC2(O)CN(C(c3c(C)nc(COC)s3)=O)C2)ccc2c(n1)NCC2 63655,N1(C(c2c(C)coc2)=O)CCC(NC(=O)CCc2c(C)noc2Cl)C2(CCC2)C1 63656,C1(C2CCCO2)(OCC(=O)NCC2CC=CC2)CCCC1 63657,C1(N(C(=O)CSS(C)(=O)=O)C)CCC(NC(c2cnc(S)[nH]2)=O)C1 63658,c1(CC)c(C(=O)NCCNC(=O)CCCc2nc(C)no2)cccc1Br 63659,c1(C(N2C(CNC(c3c(C)coc3)=O)CC2)=O)c(C)nn(CC(F)(F)F)c1Cl 63660,Cc1nsc(CNC(=O)C=CC(C)NC(C2(CO)CCOC2)=O)n1 63661,N1(C(C)=O)CC(N=c2[nH]c(=N)[nH]c(=NC(C)CCc3ccc(C)cc3)[nH]2)C1 63662,C1(NC(c2nc(C)c(C)s2)=O)CCCN(C(=O)CN2C(C)CCC2C)CC1 63663,S(=O)(=O)(c1ccc(=NCCC2CCSC2)[nH]c1)NC1CC(C)(C)SCC1 63664,Cc1cc(C(=O)NCC2COC(CNC(=O)CCc3n[nH]c(=N)s3)C2)nc(O)n1 63665,CC1N(C(=O)N(c2ccc(F)cc2F)C2CCCO2)CCC1(C)C 63666,C=C(C)CC(C(=O)N(C)C)NCc1cn(C2C=CCC(C(=O)OC)C2)nn1 63667,N1(C(C(N2CCCCC2=O)C)=O)CCC(F)(CNC(c2cn(CCO)nn2)=O)C1 63668,c1(C(=O)OCC(=O)N(C(CC)CC)C2CC2)cc(Br)c(C)s1 63669,N1(C(CC2(COC)CC2)=O)CC(CNC(c2cc(OC)nc(F)c2)=O)C(C)(C)C1 63670,c1(NC(C)=O)cccc(F)c1NC(=O)COc1ccc(F)c(F)c1 63671,CC1CC(C)(CN2CC3CC2(c2cn(-c4cccc(C5CC5)c4)nn2)C3)CCO1 63672,CC(C)C(O)C(=O)NC(C)(CNC(=O)C(C)(C)C1CCOCC1)C(C)C 63673,Cc1conc1C(=O)NC(C)C(c1ccccc1)NC(C1CSC1)=O 63674,CC(=O)CCCCC(=O)N1CC=CC1(C)C(=O)NCC(C)CC(F)(F)F 63675,C1(C)(C(N2CCC(O)(C(C)CNC(c3ccc(CO)o3)=O)C2)=O)CCC2CC2C1 63676,c1(CC(=O)NCC2(C)CCN(C(C3(CO)COC3)=O)C2)ccc(S(N)(=O)=O)cc1 63677,C1(NC(C2COCCO2)=O)CC(C(N2CCC(CCO)CC2)=O)C12CCC2 63678,C12(C(=O)NCC(C)(C)CNC(C3(C)CCOC3)=O)CCC(CC1)C2(C)C 63679,CC1CCC(O)CN1Cc1nc(Cc2cccc(Cl)c2)no1 63680,N1(C(C(CCSC)O)=O)CC(C(=O)NC2CCCC2N=[N+]=[N-])CC(C)(C)C1 63681,c1(CC)cnc(Cl)cc1NC(c1cc(C(C)=O)n[nH]1)=O.C12CC3CC3N1C2 63682,c1(C(N(C2CCCC(NC(CCC=CC(C)C)=O)C2)C)=O)cc(Cl)cc(F)c1F 63683,c1(CNC(C(=O)NC(c2nc(C3CCCCC3)no2)C)=O)cccc(F)c1 63684,N1(C(C2C(CC)(Cc3ccc(Cl)cc3)NCCC2)=O)CCC2(CC1)CN(C)C2 63685,C(C(C)(C)CC(=O)N1CCC(C)C(C)C1)NC(COCCCOC)=O 63686,N1(CC2N(C)CCCC2)CCC(NC(=O)Cc2ccc(F)cc2F)C(C)(C)C1 63687,CCCCCCCCC(C)CC(=O)N1CC(NC(=O)CCNC(=O)OC)C(C)C1 63688,CN1CCN(CC(=O)NCCOCC(F)(F)C(F)F)CCC1=O 63689,C1(=CC(=O)NC2(CNC(C(C=C)C)=O)CC2)CCC(C)CC1 63690,C(CCCCCC(=O)N1CCC1c1ccccc1CC)n1cc(CCCC)nn1 63691,N1(CC)CCCC(C(=O)NCC2CN(C(=O)COC)CC2C(F)(F)F)C1 63692,Cc1noc(C(C)C)c1C(=O)NCC(C)(C)CCNC(C1(N(C)C)CCC1)=O 63693,c1(C(=O)NC(c2ccccc2C(F)(F)F)C=C)ccc(I)c(OC)c1 63694,c1(SC)ccc(Cl)c(C(=O)NC2CN(C(=O)CN(C3CCC3)C)CCC2CO)c1 63695,C1(NC(CC2(CNC(C(CC)C)=O)CC2)=O)CC2CCCCCC12 63696,N1(C(c2c(C)snc2)=O)C(C(=O)NCC2CCOC2(C)C)CC2CCCC12 63697,C1(CNC(c2c(C)nc(C(C)C)o2)=O)CN(C(C23CC(CO2)C3)=O)CCC1(F)F 63698,Cc1cc(CC(=O)N(C(C)CNC(=O)CC2CCC(=O)CC2)C)n(C)n1 63699,N1(C(c2c(SC)snn2)=O)CC2CC(CNC(C3CC4(CC4)CO3)=O)C2C1 63700,C1(CNC(N2C(C(=O)OC)CCC2c2ccccc2)=O)CCC(OC)CC1 63701,Cc1nc(=N)[nH]c(=NCCCC(C)NC(C2CC3CCC2CC3)=O)[nH]1 63702,c1(COC)nc(N2CCC(C)C2CNC(=O)CSc2cccc(Cl)c2)cc(Cl)n1 63703,c1(C(CC)=O)cc(C(=O)NC(C)C(C)NC(=O)CCn2cccnc2=O)ccc1F 63704,N1(C(C(C=C)(C)CC)=O)CC(C2CCCN(C(c3ncn4ccccc34)=O)C2)C1 63705,c1(CN(C(C2CCN(C(c3csc(CO)n3)=O)C2)C)C)cnc2[nH]cncc1-2 63706,C(=O)(C1=NOC2(CCOC2)C1)N1CCC(CN(C(=O)CSCC(N)=O)C)C1 63707,CCCCCC(O)C(=O)NCC1CC(F)(F)CN1C(=O)CC(C)CCC=C(C)C 63708,c1(CC)cnc(C(=O)N(C2CCN(C(C3COCC3(C)C)=O)C2)C)nc1 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63796,C1(N(CCOCCN(C(CCOCCN(C)C)=O)C)C)CCN(C)CC1 63797,N1(C(c2nc(CC)sc2)=O)CC(C)C(NC(c2ccon2)=O)C(C)C1 63798,C(=O)(C(C)(C)Oc1ccccc1)NC1CC(NC(CCSCC(C)C)=O)C1 63799,CC(C)(C)CCCC(=O)NC1CCC1NC(C1(C(F)F)CCCCC1)=O 63800,c1(C(N(CCOCC=C)C)=O)coc(C(C)NC(C2(CSC)CC2)=O)n1 63801,CCCCC(O)C(=O)NCC1(O)CCCN(C(=O)COCCC(C)C)C1 63802,N1(C(CC2(OC)CC2)=O)CC(NC(=O)Cn2nc(C)c(C)c2C)CC(F)C1 63803,C(=O)(C(=O)N=c1ncn(Cc2ccc(Cl)cc2)[nH]1)NC(C)CN1CCOCC1 63804,N1(C(C(CC)CC)=O)CC(CNC(c2ccnc(C)c2C)=O)OC2(CCC2)C1 63805,N1C2c3ccccc3OCC2CCCCC(=O)Nc2ccc(OC)cc21.OC.OC 63806,CCC(C(=O)N1CC2CCC(CNC(C34CCCC3CCC4)=O)C2C1)C(F)(F)F 63807,C1(CNC(c2cc(OC)ns2)=O)CC2CCC(C1)N2C(=O)Cc1ccccc1F 63808,n12ccc(c1)C(=O)NCC2.C1CC12CC2.C12(CC1)CC(=O)N2.CC(=O)NC 63809,c1(CNCCN(C)C)csc(=NC(CCO)C2CC2)[nH]1 63810,N1(C(c2ccc(OC)c(I)c2)=O)CC(NC(c2cnsn2)=O)CC(F)(F)C1 63811,CC(CC(=O)NC1(C)CCN(C(c2cnn(CCF)c2)=O)C1)C(F)F 63812,c1(OC)ncc(C(N2CC3CCC3(CCNC(=O)C(C)(C)C(C)C)C2)=O)cc1C 63813,Cc1ccc2c(=NCCC3CC=CC3)[nH]c(=NC(C)c3ccccc3)[nH]c2c1 63814,C1(OC)CN(C(=O)C(C)=C(C)C)CCC1NC(=O)CN1CCCCC1C 63815,c1(CNC(C=CSC)=O)ccccc1CNC(c1coc(O)n1)=O 63816,Cc1cc(C(N2CC(C(N3CC(S(N)(=O)=O)C3)=O)CC(C)C2)=O)nnc1C 63817,c12nnc(S)nc1S2.N1(C(CCC)=O)CCN(C(C)=O)CC1CC(C)C 63818,N1(C(c2c(OC)oc(C)n2)=O)CC(NC(c2ccc(C#N)s2)=O)C2(CC2)C1 63819,N1(C(c2n(C)ncn2)=O)CCCC(C2CN(C(=O)CCC3CCC3)C2)C1 63820,CC(C)(O)C(F)(F)C(=O)NC1CC(C(F)C(=O)NCCCSC(F)F)C1 63821,c1(C(N2CCC(C)(NC(CN3CCC(C)CC3)=O)C2)=O)cccc2c1COCC2 63822,c1(C(C)CO)nc(-c2cccc(N)n2)nn1CC1(C)CCC1 63823,N1(C(CCC2N(C(C3N(C4(C)CC4)CC3)=O)CCC2)=O)CCC2(COC(=O)N2)C1 63824,C1(NC(CC2N(C(C)=O)CCC2)=O)CCC(CNC(c2cnnn2C)=O)CC1 63825,C1(CC)(NC(c2ccc(F)c(C(C)(C)F)c2)=O)CCCN(C(=O)C(C)(C)OC)C1 63826,c1(C(=O)NC2CCN(C(c3ccnc(OC)n3)=O)C2)cccn2ccnc12 63827,c1(NC(C2CCN(Cc3ccncc3O)CC2O)=O)cnc(Cl)cc1[N+](=O)[O-] 63828,C(CNC(c1n[nH]c2c1COC2)=O)(CC(F)(F)F)NC(CC(C)N(C)C)=O 63829,c1(C(=O)NCC2N(C(C(C)SC)=O)CC2)ccc(S(=O)(=O)N2CCCCC2)cc1 63830,c1(CCN(C(=O)Cc2ccccc2)CCc2ccccc2)csc(C(F)(F)F)n1 63831,CCC(C(=O)N(CC(C)(C)CNC(c1cn(C(C)C)nn1)=O)C)NC(C)=O 63832,C(=O)(CCCCCC#N)N1CC(CNC(C(C)(C)SC)=O)OCCC1 63833,C1(F)(C(=O)NCC(COC)O)CCN(C(C2COCCC2C)=O)CC1 63834,C(=O)(CC1CCOc2ccccc21)N1CC(C)C(NC(=O)C=CBr)C1 63835,Cc1cccc(CC(N2CCC(C)(CCNC(=O)CC(C)(C)O)C2)=O)c1F 63836,N1(C(CCOCC)=O)CCCC2CN(C(c3ccc(CC(C)(C)O)s3)=O)CC12 63837,Cc1ccc(C(F)C(N2CCCC2C(C)(C)CNC(=O)C2CC2)=O)cc1 63838,c1(C(N2CCC(c3cn(-c4ncc(Br)cn4)nn3)C2)=O)cccc2oc(O)nc12 63839,c1(COC(c2c(C)nsc2)=O)ccc(OCc2ccccc2)cn1 63840,N1(C(c2c(C(C)C)scn2)=O)CC(CNC(C2CCCN(C)C2)=O)C2(CCC2)C1 63841,S(=O)(=O)(CCC(=O)NC1CC(C)N(C(c2ccnnc2)=O)C1)NCCNC(C)=O 63842,c1(CN(C(COC(CC)C)=O)CCNC(C2CC(C)=NO2)=O)cccc(Cl)c1 63843,C1(C(=O)NC2(CC)CC2)OCCC1NC(c1cnn(C(C)C)c1)=O 63844,C1(CC(=O)NCC(O)CNC(c2c(Cl)n[nH]c2C2CC2)=O)CCCCC(=O)N1 63845,C1(C(N)=O)CN(C(=O)C(CCF)NC(=O)CC2CC(=O)NC2=O)CC12CC2 63846,C(CC(C)C(=O)NC(CNC(C1(c2cc[nH]n2)CCC1)=O)C(C)C)=CC 63847,CCCCCC(F)C(=O)N1CC(CNC(=O)CCN2CCOCC2=O)CC(C)C1 63848,C1(NC(=O)C=Cc2nccs2)CCOC(C(=O)NCCC2CC=CC2)C1 63849,c1(CNC(C(c2ccc(Cl)c(Cl)c2)N)=O)cc(C(F)(F)F)ccc1Cl 63850,C1(NC(=O)NCc2c(C)cc(C#N)cc2)CCC2(CC1)OCCO2 63851,C12(NCC(CSC)C)CCC(CC1)NC2=O 63852,Cc1nn(C)cc1C(=O)NC1CCCC1C(=O)NCC(O)C1(Cl)CC1 63853,C1(C(N(C2CCCN(C(=O)Cc3cscn3)C2)C)=O)CCCCCCC1 63854,C1(OC)CCC(C(N2CCCC(NC(c3cnn(C)c3C)=O)C2)=O)CC1 63855,CC1CCC(O)(C(N2CC3C(C(=O)NC(CC4CC4)CO)C3C2)=O)CC1 63856,C(C)(C(=O)N(C)Cc1cccnc1)(C1CCOCC1)OC 63857,Cc1cccn2cc(C(=O)NC(C)CCN(C(=O)CN(C3CCC3)C)C)cc12 63858,Cc1nc(NC(C)(C)CN(C(=O)CSC(F)F)C)cc(Cl)n1 63859,c1(C(=O)NC(CNC(COCC=C)=O)C(C)C(C)C)cc(Cl)cc(Cl)c1Cl 63860,Cc1cnc(C)c(NC(C2(F)CC=CCC2)=O)c1 63861,C1(C(=O)NC(CC)C)CC2CCC1N2C(=O)C=C=C(C)C 63862,N1(C(C(COC)C)=O)CC2CCCC(CNC(C3CCC(=O)N(C)C3)=O)C2C1 63863,CCCCCCC(C)C(=O)NCC(C(C)C)NC(c1c(C)cnnc1O)=O 63864,c1(C(N2C(C(C)NC(C(F)=CC)=O)CCC2)=O)ccc(Br)c(SCC)c1 63865,Cc1scc(C(=O)NC2CN(C(c3cc(CO)[nH]n3)=O)CC2CC(C)(C)C)c1C 63866,CC(C)C(C(=O)NC1(C)CC2(CCC2)C1)C(C)NC(c1cc(C#N)ccc1N)=O 63867,N1(C(C(COC(C)C)NC(C)=O)=O)CC(N(C(=O)CCn2cnnn2)C)C(O)C1 63868,C(=O)(C1=Cc2cc(Cl)ccc2OC1)N(CCN(C(C1C(C)C1C)=O)CC)CC 63869,c1(OCC)cccc(CC(=O)NC2CC2CNC(=O)Cc2ccnc(OC)c2)c1 63870,N1(C(CSCC(N)=O)=O)CC2CCCCC2(CNC(=O)C=C2CCCCC2)C1 63871,c1(OC)cc(Cl)ccc1C(N1CCC(O)C(F)C1)C(=O)NC(c1ccccc1)C 63872,Cc1nccnc1C(N1CCC(C(F)C(=O)N(C)CCN2CCCC2)C1)=O 63873,C1(CC(NOCC#C)=O)CC(NC(C2CCN2CC)=O)C1(C)C 63874,C1(C(C(=O)NCCCOC=C)NC(=O)CCn2cccc2)CC=CCC1 63875,c1(CC(=O)NCC(CNC(COCC=C)=O)(C)C)cc(Cl)cc(Cl)c1 63876,C1(CC(N2CC(SC)C(NC(=O)Cc3cc[nH]n3)C2)=O)CSc2ccccc2O1 63877,N1(C(=O)Nc2c(C)cc(N3CCOCC3)cc2)CCN2CCOCC2C1 63878,Cc1ccsc1CC(=O)NCCC1CC(NC(c2nocc2C(C)C)=O)C1 63879,C1(C(NOCC(CC)C)=O)CCC(O)CN1C(C1CCCC(C#N)C1)=O 63880,N1(C(c2n(CC)ncc2)=O)CC(C(=O)NCC(C)OCCO)CC12CCC2 63881,C1(C(F)(F)F)(C(=O)NCC(CC=C)NC(C2(n3cccn3)CC2)=O)CC(C)(C)C1 63882,c1(C(N2CCC3(CN(C(c4cc(C)ns4)=O)C3)C2)=O)cn2cccc(F)c2n1 63883,O=C(C1=Cc2ccccc2OC1)NC1CN(C(c2n[nH]cc2Cl)=O)CC12CCC2 63884,C(=O)(CC1CCOc2ccccc21)N1CC(NC(CSSC)=O)C(C)C1 63885,C1(C(=O)NC(C2CN(C(C3COC(C)C3)=O)CCO2)C)(OC)CS(=O)(=O)C1 63886,C(c1ccc(F)c(Cl)c1)=CC(=O)NC1C(C)CN(C(=O)CN2CCCNC2=O)C1 63887,C(CCCCC(=O)N1C(C(=O)N(CCO)C2CC2)CCC12CC2)OC 63888,CC1CC(C(=O)NC(c2cnn(C)c2)C(=O)NCCN2CCCNC2=O)CCS1 63889,CN1CC(NC(c2ccc(-c3cscn3)nc2)=O)Cc2ccccc21 63890,CCC(C(=O)NC1CC(N(C(=O)COC2CCCOC2)C)C1)C(C)(C)CC 63891,c1(C(C)C)cc(=NCCC2CCN(C(C3CCCC(F)C3)=O)C2)[nH]c(Cl)n1 63892,c1(OCC)cc(CNc2ccc(C(=O)NC(C)(C)C)o2)ccc1O 63893,c1(C(c2nnnn2C)N(C(C)C)C(C)C)ccc(CN(C)C2CC2)cc1 63894,S(=O)(=O)(C1CCNC(C)(C)C1)Nc1cc(C)cc(C(F)F)c1 63895,N1(C(C=C(CC)CC)=O)CCC2CCCC12C(N1CCCC1CSC)=O 63896,C1(CC)CN(C(c2c(Cl)cccc2Cl)=O)CCN1Cc1cccc(I)c1 63897,C(=O)(CCCCCNC(C1CC(C)(F)C1)=O)NCCCOCCCC 63898,c1(CC)ncccc1S(C)(=O)=NC(=O)C1(Cl)CC12CCC2 63899,C1(C)(C(=O)NC(c2n[nH]c(=N)s2)C)CC12CCN(c1cccc(C3CC3)n1)CC2 63900,Cc1c(C(N2CCC(F)(CNC(=O)C(C)n3cnnn3)C2)=O)ccc2n[nH]cc12 63901,c1(C(N2CC(NC(CCCOC(C)=O)=O)C(O)C2)=O)ccc(OC(F)F)nc1Cl 63902,CC1CN(C(C2CC23CCSCC3)=O)CCN1C(=O)CCCC1CCCCC1 63903,C=CC(CC(=O)NC(C)CCCCNC(c1cc(OC)no1)=O)c1ccccc1 63904,C1(N(C(=O)COC(F)(F)F)CC#C)CCN(C(C2CC2c2ccn(C)n2)=O)CC1 63905,N1(C(C2(C)CC=CCO2)=O)CC(CNC(=O)Cc2cscn2)C2(CCC2)C1 63906,C=CCCC(CC(C)C)C(=O)N(CCNC(=O)C(C(C)C)NC(=O)OC)CC 63907,C1(N(C(C(=O)NCC=C)C)C)CCN(C(C2C(=C)C2C(=O)O)=O)CC1 63908,C1(CC=C)(C(N2CCCCC2CC(N)=O)=O)CCCN1C(C1CC2CCC2C1)=O 63909,Cc1n[nH]cc1C(=O)NC1(C(=O)NC2CC2CN(C)C)CCC1 63910,C1(CC)CN(C(c2cc(C3CC3)cnc2Cl)=O)CCN1C(=O)C(C)OC 63911,C(=O)(C1=C(Cl)CCC1)N(CCOCCCN(C)C(C1COCC(C)(C)O1)=O)C 63912,c1(NC(CC)CSC)cc(=NCC(Cc2ccccc2F)CO)[nH]c(C)n1 63913,CC1CC(C)CN(C(=O)CNC(=O)NCCCN(C)CCN(C)C)C1 63914,C1(C(=O)NCC(CC=C)NC(C2(CCOC)CCCC2)=O)CCCC2(CC2)C1 63915,n1(CC(=O)NC2C(C)CN(C(=O)CN3CC=CC3)C2)ccc([N+](=O)[O-])n1 63916,Cc1ccc(C(=O)N(CCC(C)NC(c2cnn(CC(C)C)c2)=O)C)cc1F 63917,CN1CCC2(CCN2C(c2ccc(-c3cc[nH]n3)o2)C(=O)NC2CCOC2)C1 63918,N1(S(C)(=O)=O)Cc2ccccc2CC1CC(=O)NCc1cc2c(s1)CCSC2 63919,Cc1cnc(C(=O)N(C2CCN(C(c3cc(Cl)ccc3Cl)=O)CC2C)C)c(C)c1 63920,CN1CCC(NC(=O)CC(C)(C)C)C12CCCN(C(C1(O)CCCCCC1)=O)C2 63921,C1(NC(CCNC(N)=O)=O)CCOC12CCN(C(=O)CC1CCC(=O)C1)CC2 63922,c1(N(C)CC2N(C(CC(CCCC)CC)=O)CCC2)nc2cc(F)c(F)cc2s1 63923,N1(C(C2CCC(=C)CC2)=O)CC2(CCC2NC(c2cc(C(C)C)cnc2O)=O)C1 63924,c1(OC)ccc(F)cc1C(=O)NC1CCCN(C(=O)CC2OCCO2)C1C 63925,c1(C(N2CC(COC)(CNC(=O)CCCF)C2)=O)cnn2ccncc12 63926,CCC(C)(C)C(=O)NCC(C)(CO)NC(c1cnc(-n2cccn2)cn1)=O 63927,N1(C(C2(N(C)C)CCCC2)=O)CC(CNC(c2csc(=N)[nH]2)=O)C2(CC2)C1 63928,c1(OC)ccc2c(CC(N3CCC(CCNC(=O)C(C)CSC)C3)=O)coc2c1 63929,N1(C(CCNC(c2cncnc2)=O)=O)CC2CC1(CNC(C1CC(F)(F)C1)=O)C2 63930,c1(NCC2C(NC(c3cnn(C)c3C3CC3)=O)CCC2)ncc(Br)cc1[N+](=O)[O-] 63931,c1(CC(=O)NC2CN(C(C3CCCC4CC34)=O)C2)ccc2c(c1)OCCO2 63932,C1(CNC(c2cc(C3C(C)C3)on2)=O)CCN(C(=O)Cc2ccn(C)c2)C12CC2 63933,C(=O)(CCN(C(=O)CCNC(=O)COC)C)NC(CNC(=O)NC)C 63934,C=Cc1ccc(C(N2CCC(NC(c3ccccc3CC(C)C)=O)CC2)=O)cc1 63935,c1(CC2(C(=O)OC)CN(C(C3(c4cccs4)CC3C)=O)C2)ccc(Cl)cc1 63936,N1(C(C2N(C(c3cc(C)ncn3)=O)CCC2O)=O)CC2CCC(O)C2C1 63937,C1(C)(CNC(CCOCC#C)=O)CCCN1C(=O)Cc1cn(C)nn1 63938,c1(C(=O)NCC2N(C(c3c(OC)c[nH]n3)=O)CC2)[nH]c(-c2cccc(C)c2)nc1C 63939,C(c1ccc(F)c(F)c1)=CC(N1C2CN(C(c3cc(OC)ncc3)=O)C(C2)C1)=O 63940,N1(CC(CNC(=O)Cc2cc3c(s2)CCC3)O)CC2CCCC2C1c1nn[nH]n1 63941,N1(C(C(CCSC)OC)=O)CCC2(CC1)CCN(C(C1(CO)CCCC1)=O)CC2 63942,S(=O)(=O)(c1c[nH]c2ncccc12)NCC(N1CCC(NC(C=NOC)=O)C(C)C1)=O 63943,N1(C(C(C)S(N)(=O)=O)=O)Cc2ccccc2C1CNC(C1CC2(C1)CC(O)C2)=O 63944,N1(C(CC2N(C)CC2)=O)CCCC(c2cc(C(c3ccco3)=O)n[nH]2)C1 63945,C1(N(c2ccc(F)cc2)C(=O)C(F)CC2CN(C(C)=O)C2)C2CCC(C2)C1C 63946,c1(C(CO)CNCC(O)CC2CCOCC2)ccc2c(c1)OCCO2 63947,C12(C)CCCN(C1)C2=O.c1(OCC)cc(COC)on1.N12CC(C1)OC(C)(C)C2=O 63948,c1(NC(c2cnc(C)s2)=O)cnc2n1CCN(C(=O)COc1ccc(O)cc1)C2 63949,c1(NC(C2C(C)C2)=O)cnc(F)cc1C(N1CC2CC2C1C#N)=O 63950,C1(NC(C2C(C)C2)=O)CC2(CCCCN2C(=O)C=Cc2ccnn2C)C1 63951,C1(C(=O)NCCC2(O)CN(C(CCOC)=O)C2)CC2CC(C1)CC(F)(F)C2 63952,C1(C(=O)NC2CC(CNC(C3(c4ccn(C)n4)CC3)=O)C2)CC2(C1)CC2F 63953,N1(C(C(C)CC(N)=O)=O)CCC2(CCCC2CNC(=O)Cc2cccnc2)CC1 63954,CN1CCC(C(N2CCSCC2)=O)(NC(C23CC(C#N)(C2)C3)=O)C1 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63972,N1(CCC)CC(C(=O)NCC2CCN2C(c2ccc(C(F)(F)F)nn2)=O)CC1=O 63973,c1(C(N2CC(CNC(c3ccoc3)=O)C3C2C3)=O)ccc2snnc2c1 63974,C1(C(=O)NCCCC(C)(C)NC(=O)C=Cc2cscn2)CCC2(CCOC2)O1 63975,C12(C(=O)NC(C3CN(c4nc(C5CCCC5)ns4)CCO3)C)CCC(CC1)CC2 63976,C(=O)(CC(C)C(F)F)NCC1(CCNC(COCCC#C)=O)CC1 63977,c1(CC(=O)NC(C(C)(C)NC(C(CC)C#N)=O)C)ccc(Br)c(OC)c1 63978,N1(C(C(C)=C2CC2)=O)CC2CCCC2(CNC(=O)C(c2ccccc2Cl)(C)C)C1 63979,c1(C(C)N(C(=O)CCCC(c2ccccc2)O)CCO)ccccc1Cl 63980,C=CC1(CC(=O)NC(C)CNC(=O)C(O)CSC)CCCCC1 63981,C1(C(=O)NC(C(C)C)(C)CNC(=O)CC(=O)N(C)C)CC2C(C1)C2(F)F 63982,C1(NC(c2cn(C3CC3)nn2)=O)CCCCN(C(C2C3CC4C(C3)C24)=O)C1 63983,Cc1cn2cc(C(=O)NC3C4CCC3N(C(=O)COCC3CCCC3)C4)sc2n1 63984,c1(C(N2CCN(C(C3(O)C(C)(C)C3)=O)CC2)=O)ccnc2[nH]c(O)nc12 63985,c1(C(=O)NC(CC(C)=O)C(=O)OC)cc2n(c1)CCSC2 63986,C(C)(CC(=O)NCC1(NC(c2ccc(Br)cc2)=O)CCC1)(C(F)F)N(C)C 63987,C(=O)(CC(C)CC(C)(C)C)N1CCC(NC(c2c(N)sc(C)c2C)=O)C1 63988,c1(CC)cc(N)ccc1C(=O)NCCN(C(C1CC2CC1C2)=O)C(C)C 63989,N1(C(CS(CC)(=O)=O)=O)CCC(C)N(C(=O)C(N2CCCCC2=O)C)CC1 63990,C1(NC(c2cc(-c3nc(C)sc3)sc2)=O)CCC(NC(c2ccn(C)c2)=O)CC1 63991,C1(NC(COCC#C)=O)CN(C(C2CCCC(O)C2)=O)CC2(CCC2)C1 63992,c1(NC(C(=O)NC(COCC)CO)=O)ccc(C)c(O)c1 63993,C#Cc1cccc(C(=O)NC2(c3cccc(Br)c3Cl)CC2)c1Cl 63994,C(=O)(C#CC1CCOCC1)NC(C1CN(C(C2CCc3nnnn3CC2)=O)C1)C 63995,c1(C(N2CC3(C(NC(c4cn5c(n4)CCC5)=O)CC3)C2)=O)c(F)ccc(F)c1Cl 63996,C1(C(N(CC)Cc2ccncc2)=O)CCN(C(=O)CCC2(C)N=N2)C1(C)C 63997,C(C(=O)NC(CNC(c1cn[nH]c1)=O)C1CC1)(C1CCCC1)OCC 63998,c1(NCCOC)nc(OC2(C)CCOCC2)cc(=NCCN2CCCC2=O)[nH]1 63999,c1(CC(=O)NCC2N(C(C3C(C)C3C)=O)CC=C2)ccc2[nH]ccc2c1 64000,C#CCC(CC(=O)OC)NC(C1CCC(C(C)C)N1C(=O)C=CCSC)=O 64001,N1(C(C(CSCC)NC(=O)CC2CCCC(=O)N2)=O)CCc2ncn(C)c2C1 64002,C1(CNC(Cc2c(C)nc(S)s2)=O)COCCN(C(C23CCC2C3)=O)C1 64003,C1(CC(=O)NC(=O)OCCc2ccnc(C(C)(C)C)n2)CCCNC(=O)C1 64004,c1(C(=O)NC2C(NC(c3c(C)ncs3)=O)CCC2)ccc(OC(C)C)nn1 64005,C1(CC=C)(C(N2CCN(C)CC2)=O)CCN(C(=O)CCCc2ncco2)C1 64006,N1(C(CNC(CC(C)C)=O)=O)CC(CC(=O)NC2CCCC2N=[N+]=[N-])CC1(C)C 64007,C1(OCCCNC(CC2(C#N)CC2)=O)CCN(C(C23CCCCC2C3)=O)CC1 64008,c1(C(=O)NCC(C)CNc2cnc(C#N)cn2)ccc(C2CC2)cc1F 64009,N1(C(C(=O)NCCCC)C)CC(C(C)OC)(OCCSCC)C1 64010,N1(C(C=C(CC)C)=O)CCC2CCC12CNC(c1ccnn1C)=O 64011,C12CC=C(C(=O)N3CC(C3)ONC1=O)C2.CCC(O)C(=O)O.C(=O)(CC)OCC 64012,c1(CC(N2CC(NC(c3cc(C(C)=O)sc3)=O)C(C)C2)=O)cccc(Cl)c1Cl 64013,c1(C(N2CCc3nc[nH]c3C2)=O)cccc2occc12.CCCC1CC(=O)N1 64014,CCC(F)(F)CC(=O)NC1CN(C(=O)C=CCF)CC1C(F)F 64015,N1(C(C(CCC)CNC(c2cc(CO)on2)=O)=O)CCOCC(F)(F)C1 64016,C=CC(CC)CC(=O)N1C2CCC1C(NC(=O)CS(C)(=O)=O)C2 64017,C1(CCOC)(NC(c2nc(C)nn2C)=O)CCN(C(=O)COCC(F)F)CC1 64018,N#CC1CN(Cc2ccc(F)nc2F)CC1NC(c1ccc(OCF)cc1)=O 64019,Cc1ccc(F)cc1C(=O)C(=O)N(C1CCN(C(C2(C#N)CC23CCC3)=O)C1)C 64020,CC1CCN(C(=O)C(=O)NC(=O)CCCC(F)(F)C(F)F)CC1 64021,c1(C(=O)NC(CNC(COCCOC)=O)C2CCC2)cc2c(s1)CC(C)(C)C2 64022,C1(C(=O)NCC(C)N(C(=O)CC2CC(=O)NC2=O)C)CCCOC1c1ncc[nH]1 64023,c1(NC(=O)NCC2(CNC(C=CS(CC)(=O)=O)=O)CC2)ccn2cc(C)nc2c1 64024,c1(N(C)CC)ccc(CCCCNC(=O)NCc2ccccc2OC)cc1 64025,c1(CC(=O)NCC2C(NC(Cc3c(C)ccnc3)=O)CCC2)c(C)cccc1F 64026,c1(C(N2CC(CNC(CC=CCC)=O)C(OCC)C2)=O)cc2c(s1)CC(C)(C)C2 64027,N1(C(C(=O)N(c2ccc(Br)cc2)C(C)C)=O)CC2(CO)CCCC2(F)C1 64028,c1(C(N2CC(SC)C(NC(c3cccn3C)=O)C2)=O)n[nH]c2ccc(Cl)cc12 64029,C(=O)(C1=CC2C=CC1C2)N1CC(NC(=O)CC2CC2)C(CO)C1 64030,c1(COC)nc2n(n1)CC(NC(c1cccc(C(N)=O)n1)=O)CC2 64031,C(=O)(CC(C(C)C)c1ccccc1)N1CC(O)(CN(C(c2c(C)c[nH]n2)=O)C)C1 64032,N1(C(CN2CCC(OC)C2)=O)CC=C(C(=O)N2CC(CN=[N+]=[N-])C2)C1 64033,C1(C2(O)CCN(c3nc4cccc(F)c4o3)CC2)(NC(=O)COCC2CC2)CC1 64034,C12(C(=O)NCC3N(C(=O)CC4CC4)CC=C3)CC3CC(C1)CC(O)(C3)C2 64035,c1(CC(=O)NC(C2(O)CCN(C(=O)C3=CSCS3)C2)C)cn2cc(F)ccc2n1 64036,Cc1nc(-c2cccnc2)[nH]c1C(=O)NCC1CC(NC(C2CCCN2C)=O)C1 64037,c1(C(N(CCOC)CCNC(=O)C(C)SC(F)(F)F)=O)ccoc1Cl 64038,C(=O)(C1=CC2C=CC(C1)C2)N1C(C(=O)Nc2cccc(CC)c2)CC1 64039,C(=O)(CC1COc2cc(O)ccc21)N(CC(C)NC(=O)CCC(=O)NN(C)C)C 64040,N1(C(=O)COCCF)CCC2(CC1)CCN(C(=O)CC1CCC13CCC3)C2 64041,N1(C(C2=CCCN(C(CC#N)=O)C2)=O)CCC2(CCC2)C(O)C1 64042,c1(C(N2CCC(N(C(COCCC=C)=O)C)C2)=O)ccn2cc(C)nc2c1 64043,N#CC1(CC(=O)NC2CCCCN(C(=O)C(F)CC3CCCC3)C2)CCOCC1 64044,c1(NC(=NC)N(C)C)ccc(O)c(Nc2cccc(C)c2C)c1 64045,N1(C(C(Cc2ccoc2)NC(c2c[nH]c(=N)o2)=O)=O)CCN2C(=O)NCC2C1 64046,C1(C(=O)NCC(CC)(C)NC(c2csc(-c3ccccc3)n2)=O)CC2CCC1O2 64047,C=CC(CC)CC(=O)NCCC1CC(OC)CN1C(=O)Cc1cc[nH]c1 64048,N1(C(C(C)C)=O)CCC(O)(C2CCN(C(c3ccc(C(C)F)cc3)=O)CC2)CC1 64049,CCC(C)C(C)CN=c1nc(N(C)Cc2cccc(Br)c2)c2sccc2[nH]1 64050,C1(C(N(C2(C(=O)NC(C(=O)NC)C)CC2)C)=O)C(C)(C)C1(C)C 64051,Cc1cn2c(CCC(=O)NCC3CC3CNC(=O)Cc3ccccc3)csc2n1 64052,CC1CN(C(=O)CC2CCC(=O)NC2)CCC1CNC(C1CC2(C1)CC(F)C2)=O 64053,Cc1cc(=NCC2CCN(C)CC2)[nH]cc1S(=O)(=O)NC1CC(CF)C1 64054,CC1(NC(c2cc(C3CC3)no2)=O)CCCN(C(c2cc(C#N)c[nH]2)=O)C1 64055,N1(Cc2nc(C)on2)CC2C(C(=O)NC(C)Cc3ccccc3F)C2C1 64056,C1(C)(OC)CCCN(C(=O)C(C)Cc2ccc(Cl)cc2)C1.C1C(=O)NCCS1 64057,c1(CC)nc(C)c(C(=O)NCC2CC(C)N(C(C3CC(OC(C)(C)C)C3)=O)C2)s1 64058,C1(C(=O)NC2(CC(=O)NC(c3ccc(C)nc3)C)CC2)CCC2(CCC2)O1 64059,c1(NCC(=O)NCCC2CC(C(=O)NCC3CC3(Cl)Cl)C2)nccs1 64060,N1(CC(C(CC)C)C)CCC2(CC1)CC2(C)C(N1CC(C(=O)OC)C(O)C1)=O 64061,c1(NC(CC(C)N(C)C(=O)NCCOC2CC2)=O)ccc(S(C)(=O)=O)cc1 64062,Cc1ccc(C)c(N(C(c2scnc2Cl)C(=O)NCC2CC2)C)c1 64063,CC(C)(C)CCCC(=O)NCC12CN(C(C3CCCN3C3CC3)=O)CC(F)(C1)C2 64064,CCC(CC)C(F)C(=O)N(C1CN(C(=O)CC(C)N(C)C)CC1(C)C)C 64065,C#CCC(C)(C)C(=O)NCC1(NC(C2CC2c2cccs2)=O)CCCCC1 64066,CCC(CC)CCC(=O)N1CC2CC1CN2C(C1(Sc2ccccc2)CC1)=O 64067,C1(NC(CN(C(=O)CCn2ccnn2)CCC)=O)CCC(C(C)O)CC1 64068,c1(CC)[nH]nc(Cl)c1C(=O)N(C)CC1(NC(=O)C(C)C2CCC2)CC1 64069,N1(CC2CCCN(CC(COC)(C)OC)C2)C(=O)NC2(CCCC2)C1=O 64070,C1(OC)CC(CNC(c2coc(O)n2)=O)N(C(C2CNC(=O)N2)=O)C1 64071,C1(NC(c2ccc(CC)s2)=O)(CO)CCN(C(c2ccnc(Cl)c2OC)=O)CC1 64072,N1(C(c2cc(COC)no2)=O)CCC2CN(C(=O)CC(F)(F)Cl)CCC2C1 64073,c1(C(N2C(C)CC(c3cn(C(C)CO)nn3)CC2)=O)cc(Cl)c2c(c1)OCO2 64074,c1(OCC(=O)OC)ccccc1NC(C1CC(C)(Nc2cc(C)c(Cl)s2)C1)=O 64075,C1(C(=O)NC2(C#C)CCCC2)CC2(CCC2)CN1C(=O)C(CCOCCO)SC 64076,c1(C(=O)NCC(CNC(Cc2c(SCC)cccc2)=O)O)cc(O)cc(O)c1 64077,C(CN=c1[nH]c(Cl)nc2c1CCC2)(c1ccccc1F)NC(c1ccc(C)[nH]1)=O 64078,C1(CNC(C(C2CC2)OC)=O)CCN(C(=O)C(C)(C)N(C)C)C1 64079,Cc1cc(=NCC2CC(C(C)C)C2)[nH]c(N2CCC(CC(F)(F)F)C2)n1 64080,C1(NC(c2ccc(SC)s2)=O)CCN(C(=O)CN2CCC(C)C2)CC1(C)C 64081,CCCCC(F)(F)C(=O)N1CC2CCOC2(CNC(C2CCNC(=O)C2)=O)C1 64082,c1(NC(=O)NC(c2ccc(NC(=O)OCC)o2)C)ccc(Cl)c(CC)c1 64083,C1(N)CCCC1(F)F.c1(CN(CC(C)(C)O)C(C2(C)CC2)=O)ccccc1 64084,C1(C(N2CC(CN(C(=O)Cc3ccn(C)n3)C)C2)=O)CCc2ccc(F)cc2O1 64085,CC(C(=O)NCCC1(O)CCN(C(=O)C(C2CCOCC2)F)CC1)C(F)(F)F 64086,N1(C(c2ccc(OC)c(Cl)n2)=O)CCCc2[nH]nc(CO)c21 64087,Cn1nc(Br)c2ncnc(NC3CCN(C(=O)Cc4nsc5ccccc45)C3)c12 64088,CC1Cc2cc(C(=O)NC3CC(F)(CNC(C4CC=CCC4)=O)C3)ccc2O1 64089,C1(CCNC(C(CCC)=CCC)=O)CCN(C(c2cc(C)nn2CC)=O)C(C)C1 64090,N1(C(C(C)NC(C)=O)=O)CC(C(=O)NC(C)C(=O)NC(C)C)(COC)C1 64091,N1(C(CCC2(C)N=N2)=O)CCCC(F)(C(=O)NC2CCN(C3CC3)C2=O)C1 64092,C1(C(=O)NC(C2CCCCC2)CNC(C2CC(OC)C2)=O)CC=CCO1 64093,N1(C(C=C(C)C(F)F)=O)CC2CC(C(=O)NCC#Cc3cccnc3)C(C2)C1 64094,N1(C(COC)=O)CC(CNC(=O)C(c2ccc(F)cc2)F)CC(C)C1 64095,c1(C(N2C(C)CCC(C(=O)O)C2)=O)ccc2nc[nH]c2n1 64096,C1(NC(CCCCCC)=O)CN(C(c2cccc(Br)c2F)=O)CC2(CC2)C1 64097,N1(C(Cc2nc(C)c(C)[nH]2)=O)CCC(C)C(CNC(c2c(C)nsc2N)=O)C1 64098,c1(OC)c(C)cc(C(N2Cc3[nH]nc(NC(=O)CCC4CCC4)c3C2)=O)cc1C 64099,Cc1nn(C)cc1C(C)C(=O)NC(c1cn(Cc2ccc(Br)s2)nn1)C 64100,N1(C(C(C)SCCOC)=O)CC2CC(C1)C2NC(=O)C(C)(C)NS(C)(=O)=O 64101,C(=O)(CCC(=O)C(C)(C)C)N1CCC(C)CC1C(=O)NC1CN(C2CCC2)C1 64102,C#CCC(O)C(=O)NCC(F)CNC(c1cccc(C)n1)=O 64103,CC(N=c1nc(C(F)(F)F)[nH]s1)C1CCCCN1C(=O)C=C1CCCC1 64104,CCC(CNC(=O)CCc1cc(Cl)cs1)N=c1[nH]c(C(=O)OC)nc(=N)[nH]1 64105,N1(C(CCC(CC)NC(c2cnco2)=O)=O)CC(C)(C)C2CCCC12 64106,C1(CC(=O)N(CCOCC=C)C)CCN(C(C2CCCCC2O)=O)CC1 64107,C(=O)(C(C)(C)CN(C)C(C1CCOC(CC)C1)=O)NC(CCC)c1ccco1 64108,N1(C(C2N(CCC)CCC2)=O)CC2CC(C)N(C(=O)CN3CCCNC3=O)C2C1 64109,C(=O)(CC(=O)N1CCCC1C(C)(C)CNC(C1CC1C1CC1)=O)NC 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64127,CC(C)(C)C(CNC(C12CC(CO1)C2)=O)NC(C1CC12CC(O)C2)=O 64128,c1(C(N2CCC(=C(Br)Br)CC2)=O)c(O)ncc2c1CCC2 64129,N1(C(C(CC#C)NC(=O)CN2CCC(=O)CC2)=O)CC2CCC=CC12 64130,N1(CC(=O)NC2CC(NC(CC(C)C)=O)C2)CCP(C)(=O)CC1 64131,N1(C(c2cc(SC)oc2)=O)C(C(=O)NCC(C)(C)C(N)=O)CCC1C(C)C 64132,c1(C(N2CC(C(C)NC(C3CCCC3C)=O)OCC2)=O)csc([N+](=O)[O-])c1 64133,N1(C(CC2CN(C)C2)=O)CC2CCC1C(NC(c1c[nH]cc(Cl)c1=O)=O)C2 64134,CCCCCC(F)C(=O)N1CC(C)N(C(c2cc(C)no2)=O)CC1C 64135,C=CC(CCC)CC(=O)N1CC(CNC(=O)C(C)(C2CC2)OC)(OC)C1 64136,N1(C(CCOCC#C)=O)CCC(NC(=O)COCCOCC)C1 64137,N1(C(C2CCCC(C)CC2)=O)CCCC2(CCCN2C(=O)Cc2cn(C)cn2)C1 64138,C1(OC)CCCC(CC(N2CC(O)(CCNC(=O)COc3ccsn3)C2)=O)C1 64139,C1(NC(=O)NCCc2sccc2F)CC[Si]2(CCCC2)CC1 64140,Cc1cc(CC(N2CC(NC(=O)CP(C)(C)=O)CCC2C)=O)cc(Br)c1 64141,C(N1CC(C)C1C1CCCO1)n1cnc(C(c2ccc(Cl)cc2)OC)n1 64142,c1(CSCC(=O)NC2C=CC(C(=O)NC(c3ccccc3)C)C2)ccc(Cl)cc1 64143,Cc1ncnc(N(C)CC2CCCCN2C(=O)C(F)CC2CCCCC2)c1F 64144,c1(OC)ccc(C(CN(C)C)NC(N2CCC(C3OCC3(F)F)CC2)=O)cc1 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64198,c1(C(N2C(C)CCC(c3ccccc3)C2)=O)cc2ccccc2oc1=O 64199,c1(OC)ccc(O)cc1C(N1CCCCC(NC(=O)C2=CCCCC2)C1)=O 64200,c1(C(N2CC(CN(C(=O)CC3CCCC3)C)C2)=O)ccn(C)n1 64201,CC(O)CCCC(=O)NCC1CCN(C(C2CN3CCC2CC3)=O)C1 64202,C1(CCNC(c2ccc(CC)o2)=O)CN(C(=O)C(c2ccc(C)o2)C)CCCO1 64203,c1(CS(C)=O)cccc(C(=O)NC2CN(C(=O)CC3C=CCC3)C2)c1 64204,C1(C(=O)NCC2(O)CCCN(C(C(C(CC)C)O)=O)C2)CC(=O)N(C)C(=O)N1 64205,C1(O)(CNC(CN(C(=O)OCC)C)=O)CCN(C(=O)C(C(C)C)n2ccnc2)C1 64206,C1(CC(C)(C)C)CN(C(C2(CCF)CC2)=O)CC1NC(=O)CSC1CCCCO1 64207,Cc1cc(CN2CC(F)(C(=O)NCc3ccc(O)cc3F)C2)ccc1F 64208,N1(C(c2cc(COC)on2)=O)CCCCC(CNC(=O)Cc2nn(C)cc2Cl)C1 64209,N1(C(C(CC)NC(C)=O)=O)CCC12CN(C(C1CCC(C(F)(F)F)O1)=O)C2 64210,C1(CC(=O)OC)Cc2ccccc2CN1C(c1cnc2c(Cl)cccn12)=O 64211,C1(CC(=O)OC(c2ncc(C(C)C)o2)C)Cc2cc(C(F)(F)F)ccc2O1 64212,c1(C(=O)NCCC2(OC)CN(C(=O)C=C(C)Cl)C2)cccc(S(N)(=O)=O)c1 64213,c1(C(N2CC(NC(C=Cc3ncc(C)[nH]3)=O)C(C)(C)C2)=O)cnc2cc[nH]c2c1 64214,c1(C(N2CCC(NC(C3CCCC3(F)F)=O)(CF)C2)=O)ccn2c(O)nnc2c1 64215,C1(N(C(c2csc(C(=O)OC)n2)=O)CC)CCN(C(=O)COC)CC1 64216,C(CNC(c1cc(C(N)=O)co1)=O)(CC(F)(F)F)NC(c1ccc(OC)nc1)=O 64217,C1(CNC(=O)CCF)CN2CCCCC2CN1C(c1onc2ccccc12)=O 64218,Cc1cccc(C(=O)NC2(C)CCN(C(C3CCCCC3C(F)(F)F)=O)C2)c1N 64219,C=C(Cl)CC(C(=O)N1CCC2(CC1)N=N2)NC(c1cccnc1O)=O 64220,c1(NC)scnc1C(=O)NC(COC)C(=O)NCCCc1cccnc1 64221,C1(CCNC(c2c(C)snc2)=O)CCCCN1C(=O)C(C)Oc1ccccc1Cl 64222,C(=O)(C(CC(C)C)NC(=O)C(C)CCOC)N(CC(CCC=C)O)C 64223,C1(NC(=O)CCc2cc(Cl)cs2)CC2(C1)CC2NC(c1cc(C2CC2)[nH]n1)=O 64224,C12(CNC(C=C(CCC)C)=O)CN(C(=O)C=Cc3ccc(C)cc3)CC(F)(C1)C2 64225,C1(S(N)(=O)=O)(C(=O)NC2CCC(NC(c3cnn(C)c3C(F)F)=O)C2)CCCC1 64226,N1(C(C(CCC)C)=O)CC(C2CCCCN(C(=O)CCC3CC3(C)C)C2)C1 64227,c1(C(=O)NCC(CN(C(C(CC)(C)C#N)=O)C)C)cccc2cccc(OC)c12 64228,c1(N2CC(C)C(CO)C2)nc2cc[nH]c2c(=NC(C)c2nnc3n2CCC3)[nH]1 64229,c1(CN2CCC(Nc3scc(C(=O)OC)n3)C2)cc(Br)ccc1C(=O)O 64230,N1(C(CC(CC(C)C)O)=O)CC2CCC1CN(C(=O)CN1CCCC1=O)C2 64231,C1(NC(CC(C)c2cccnc2)=O)CC12CCN(C(=O)C(C)(C)CCC#N)CC2 64232,C(=O)(CC1C(=O)Nc2c(F)cccc21)NCC1(NC(=O)CCF)CCOC1 64233,C1(CC(C)(C)C)CN(C(=O)C2CC2)CCN1C(C1CCC(C(=O)O)C1)=O 64234,C(=O)(CCCCCS(N)(=O)=O)N1CCC(C)C1CNC(c1cc([N+](=O)[O-])c[nH]1)=O 64235,C(=O)(C(C)CNC(=O)C(CC1CC1)NC(C1CC1C#N)=O)NC 64236,N1(C(CC2C(C)C2)=O)CC(NC(C2(C)CCCCO2)=O)C2CCCCC12 64237,C(CCCCCNC(C1CCCN1c1ccccc1)=O)NC(COCCOC)=O 64238,c1(OC)cc(CC(=O)NC2(CNC(C3CCC(C)(C)CO3)=O)CCC2)cc(F)c1 64239,CC(CC1CC1)C(=O)NC1CC(NC(=O)CCC2CC2(C)C)C1 64240,CC(CCC(C)(C)C)C(=O)N1C(C(N2CC(CO)C2)=O)CC2CC12 64241,c1(C(N(C)CC2C3CN(C(C4(N(C)C)CCCCC4)=O)CC23)=O)ccn(C)c(=O)c1 64242,CC1CCCC(CNC(c2cc(CNC(c3cc(Cl)n[nH]3)=O)nn2C)=O)CC1 64243,C1(C(=O)NCc2cccnc2O)CSCCN1C(c1ccnc(Br)c1)=O 64244,N1(C(Cc2cc(C)sc2)=O)CC=C(C(C)(C)C(=O)N2CCCCC2CC(C)O)C1 64245,c1(-c2cn(C(C(=O)NCCC)C)nn2)ccc(NC(=O)C(C)COC)c(Br)c1 64246,N1(C(CC(=O)OCC)=O)CCCC(C2CCCCN2C(c2cccn2CC)=O)C1 64247,CC1(C)C(NC(=O)CC(C2CC2)C2CC2)CC1CC(=O)Nc1cccc(OCF)c1 64248,c1(C(N2CC(C)(OCC(=O)N(C)Cc3cc(C)no3)C2)=O)ccc(F)c(F)c1 64249,C(=O)(C(CC(C)(C)C)NC(c1ccc(F)cn1)=O)N(CCCCCC=C)C 64250,N1(NC(=O)C=CC(F)(F)F)CCOCC1.C1CCNC(=O)NCC(=O)N1 64251,Cc1nn(C)cc1S(=O)(=O)NC(c1cc(N(C)C)nc(Cl)c1)=O 64252,C12(NC(c3cc(O)ncn3)=O)COC(C1)C(NC(c1scnc1Cl)=O)C2 64253,N1(C(c2cc(OCC)ncc2)=O)CC2CC(Nc3nc4ccccc4s3)CC1C2 64254,C1(C)(CNC(COC(CC)C)=O)CCCN1C(=O)CN(C1CCC1)C 64255,C(=O)(C(C(F)(F)F)C(F)(F)F)NCC1C(NC(c2cn(C)nc2C2CCC2)=O)C1 64256,C1(CNC(=O)CCCC2CCCC2)CC2CCC1N(C(c1cccnn1)=O)C2 64257,C#CCCCCCNC(c1ccc(CNC(=O)CC2CCCCC2)nc1)=O 64258,c1(C(=O)NC(C(C)C)CNC(c2cnn(C3CC3(F)F)c2)=O)cnc(N)cn1 64259,c1(C(=O)NCC(C)N(C(c2n(CCC)ncc2)=O)C)ccc2c(c1)C(=O)CCN2 64260,N1(C(C)C)CC(NC(c2cc(CNC(C3CC3(F)Cl)=O)[nH]n2)=O)CC1=O 64261,C(CC(CC)CC)(c1n(CC=C)nnn1)Nc1cccc(C(C)CC)c1 64262,c1(C(N2CC(C)(NC(C3C(OCC)C3)=O)C2)=O)ncc2[nH]ncc2n1 64263,N1(C(C(CC)SC)=O)CCC(CNC(c2cc(C(=O)OC)nn2C)=O)CC1 64264,C12(C(N3CCC(C(C)NC(C=C(C)Cl)=O)C3)=O)CC3CCC(CC(C3)C1)C2 64265,Cc1cccc2c(CN3CCC(NC(c4cnn(C)c4)=O)C(O)C3)c[nH]c12 64266,C(c1nc(C)c(C)[nH]1)=CC(=O)NCC(CC)NC(c1ncc(C)cc1O)=O 64267,C1(CNC(c2ncncc2Cl)=O)C2CCC(C2)N1C(C12CC3CC1C2C3O)=O 64268,Cc1cc(=NCC(C)c2ccsc2)[nH]c(N2CCN(C(=O)CCC(C)C)CC2)n1 64269,CCCC(CCC)C(=O)NC1CCCC(NC(c2cc(C(F)(F)F)on2)=O)C1 64270,CC1CCCCC1(C)C(=O)NCCOCCN(C(=O)COc1cncc(Cl)n1)C 64271,c1(C(=O)NCC2OCCCN(C(C3(C)COC3)=O)C2)ncnc2c1CCCC2 64272,C1(CNC(C(CC)CC)=O)CN(C(c2ccnc(C3CC3)n2)=O)CC1(C)C 64273,N#Cc1cc(C(N2CCC3CN(C(C4CCCN4N=O)=O)C3C2)=O)ccc1F 64274,c1(N2CC3CN(C(c4cc(C)nc(C)c4)=O)C3C2)ncnc2n[nH]cc12 64275,c1(CC)cccc(C(=O)NC2(CNCc3ccc(CSC)o3)CCOCC2)c1C 64276,Nc1cc(C(=O)NC2CCCCC2NC(=O)C=CCF)cc([N+](=O)[O-])c1 64277,c1(C(=O)Nc2cccc(-n3cc(C(=O)OC)nn3)c2)ncc(Cl)nc1OC 64278,C1(NC(Cc2ccc(C(C)C)cc2)=O)CCN(C(=O)C=Cc2ncc[nH]2)C(C)C1 64279,c1(CC(N2C(C(C)NC(c3c(C)cc[nH]3)=O)CCCC2)=O)c(F)cc(F)cc1F 64280,c1(C(=O)NCc2nnn(C)n2)c[nH]c2cc(C(F)(F)F)ccc2c1=O 64281,c1(C(=O)NC(CC=C)CNC(C2(OC)CCSC2)=O)cn2ccsc2n1 64282,c1(C(N2CCC(N(C(CSCC)=O)CC)C2)=O)nnc(O)c(Br)c1O 64283,C(=O)(C1=CCC(F)(F)CC1)NCC(CNC(C1C(CC)CCO1)=O)O 64284,C1(C(=O)NC2(C)CN(C(C(c3cscn3)N(C)C)=O)C2)CC2CCC(C1)C2O 64285,c1(C(=O)NCC(CC=C)NC(=O)CC)cnc2cccc(C)n12 64286,n1(CC)ccc(CC(=O)NCC(CNC(C2CC=CCC2)=O)OC)n1 64287,N1(C(CC=CCNC(C(C=C)C)=O)=O)CCN(CC)CC1 64288,Cc1cnn(C)c1CC(=O)NCC1(C)CC(NC(c2ccc(N(C)C)nn2)=O)C1 64289,c1(C(N2CCC(NC(C(C(C)(C)C)OCC)=O)(CF)C2)=O)cc(C)c(N)cc1Cl 64290,c1(NC2CC(CNC(CC(CC)C(C)C)=O)C2)ncnc2sc3c(c12)CCC3 64291,N1(C(C2CCN(C(C3CCC(CC)CC3)=O)C2)=O)CCCNC(=O)C12CC2 64292,c1(NC(C2(F)CCN(Cc3nccc(C(=O)OC)c3)C2)=O)cc(Cl)c(Cl)cc1O 64293,c1(C(=O)NC2(C)CN(C(C34CCCC3CCC4)=O)C2)cc(C#N)ccc1F 64294,C(=O)(C(COC)COC)NCC(C1CCCC1)NC(c1cc(OCC)no1)=O 64295,C1(CCN(C(C2CCN(C(=O)NC)C2)=O)C)CCCCN1C(c1ccc(F)s1)=O 64296,C1(CN(C(CN(C2CC2)CC)=O)C)CCCCN1C(=O)CC1CCOC1(C)C 64297,N1(C(C(CSC)OC)=O)CCC2(CCC(NC(c3[nH]c(O)nc3C)=O)C2)CC1 64298,C(CCCC(C)(C)C)NC(CC(CNC(C1CC1(C)C)=O)OC)=O 64299,Cc1nn(C)c(C)c1C(=O)NC12CC1CN(C(=O)CC1CCC(C)(C)CO1)C2 64300,c1(COC)nc(NCc2cnn(CCF)c2)cc(=NC(C)C2CCCO2)[nH]1 64301,C(=O)(CC1=CCCCC1)NCC1(COC)N(C(C2(CCCC)CC2)=O)CCC1 64302,C1(NC(c2cc3c([nH]2)CCCC3)=O)CCN(C(C2(O)COC2)=O)CC12CCC2 64303,C1(NC(COCCCC)=O)CC2CCC(C1C)N2C(c1cnn(CCF)c1)=O 64304,C(N=c1[nH]c2c(c(=NCc3cccc(C#N)n3)[nH]1)COC2)C1CCCC(C)CC1 64305,CCC(CC(=O)NCC1C=CCN1C(c1cc(OC)cs1)=O)C(C)C 64306,Cc1nc(C(=O)N(C)CC2CCCCN2C(C2CC2c2cn[nH]c2)=O)c(C)s1 64307,C1(C(N2CCC(NC(C3CCOCC3)=O)C2)=O)(OCC)CCOCC1 64308,CCC(F)(F)C(C)(C)NC(=O)C(O)CNC(c1cc(COC)no1)=O 64309,c1(C(=O)NC2CCN(C(C3NC(=O)OCC3)=O)C2)ccc2nc(O)[nH]c2c1F 64310,Cc1cccc(Br)c1C(C(=O)NCC1(O)CCCOC1)NC(=O)CCC1(C)N=N1 64311,c1(C(=O)NCCC(C)(C)NC(C2C(C)OCC2)=O)ccc(C(F)(F)F)cn1 64312,CC1(C)CCCN(C(=O)Cc2n[nH]cc2Br)C1CNC(c1scnc1Cl)=O 64313,CCC(CN(C)C)CC(=O)NC1(CO)CN(C(C2CC(OC3CC3)C2)=O)C1 64314,c1(CC(=O)NC2CCCC(NCC3(C)CC3)C2)ccc2ccccc2c1 64315,C1(NC(C2(CC)COC2)=O)CCC2CCN(C(c3csc(=NC4CC4)[nH]3)=O)C1C2 64316,N1(C(C(C)CNC(C2CCCN2C2CC2)=O)=O)CCCCC(CO)C1 64317,N1(C(C(C)SC)=O)CC2(CCCC2)C1C(=O)NCCc1ccccc1 64318,C(c1ccc(OC)cc1OC)=CC(N1CCCC(NC(CCOC)=O)C1C)=O 64319,C(=O)(C(C)(C)COCC)N(CC(=O)NC(C=C)CO)CCOC 64320,C1(N(C(CCOCCOC)=O)C)CCN(C(c2cnn(C)c2N)=O)CC1C 64321,N1(C(=O)COCC2CCOC2)CC2(C1)CN(C(=O)C(F)C1CCC1)C2 64322,C1(NC(Cc2n(C)ncc2)=O)CC2CN(C(c3ccn(C(C)(C)C)n3)=O)CC12 64323,N1(C(C(COC(C)=O)(C)C)=O)CC2(CO)CC1(C(=O)N(CCCN(C)C)C)C2 64324,C1(F)(CNC(C2N(C)CCC2)=O)CCN(C(c2ccc(-c3cccs3)o2)=O)C1 64325,C1(CNC(C(C=CC)O)=O)CC2COCC2N1C(=O)CC1CCC2CC2C1 64326,c1(C(N2CC(CNC(C(C=C)(C)O)=O)C(F)(F)CC2)=O)ccc2nc(O)[nH]c2c1 64327,N1(CCNc2cn(CC)nc2)CCCCC1CC1CC1 64328,C(=O)(C(F)C(C)(F)F)NCc1cc(C(N2C(C)(CCC)CC2)=O)no1 64329,N1(C(c2cc(C)oc2C)=O)CCCOC(CNC(=O)Cc2cocn2)C1 64330,C1(CNC(c2n(CCCC(=O)OCC)nnn2)(C)CCI)COC(C)(C)O1 64331,CCC(CC)C(F)C(=O)NCCCC(O)C(=O)N(C1CC1)C(C)C1CC1 64332,C12(NC(C(C)CC3CC3)=O)CCCC1CN(C(=O)Cn1ccc(C3CC3)n1)C2 64333,Cc1cc(C=CC(=O)NCC(C)(O)CNC(=O)C(C)Cc2ccco2)c[nH]c1=N 64334,C(=O)(C(O)CCN(C)C)NC(C(N1C(C=C)CC1)=O)(C)C1CCC1 64335,c1(CNC(C(C)=C(CC)C)=O)ccccc1CNC(=O)COC1CCCOC1 64336,CCC(CC(=O)N(CCCN(C)C(C1(C)CCNC1=O)=O)C)C(=O)OC(C)(C)C 64337,N1(C(Cc2scc(C)n2)=O)CCCC(C)C1CCNC(=O)CCc1cncn1C 64338,c1(C(=O)NC(C(=O)NCCN(C(=O)CNC2CC2)CC)C)cc(Cl)ccn1 64339,c1(C(N2CC3C(NC(C(C(C)(C)F)(C)F)=O)C3C2)=O)ccc(N)c([N+](=O)[O-])c1 64340,C(=O)(CC(CC)C(C)C)N1CCN(C(c2c(NC)nsn2)=O)C(c2ncc[nH]2)C1 64341,N(C1CC(C)n2ncnc21)CCC(=O)NC(C)Cc1ccccc1 64342,C(CCCC(=O)NC1CCCC1NC(=O)Cc1ccc(C)o1)OC 64343,c1(SC)nc(N(C(C)CCNC(=O)C(CO)NC(N)=O)C)cc(Cl)n1 64344,CN1C(=O)OCC1C(=O)NCC12CC1CN(C(=O)CCC1CC(F)(F)C1)C2 64345,C(C(CC(F)(F)F)NC(=O)CCc1nccs1)NC(=O)C=CCO 64346,C(c1cocn1)=CC(=O)NCC1(C(=O)NCC2(C(C)(C)C)CCC2)CC1 64347,c1(CC)cc(C(=O)NCCCNC(c2cnncc2C(C)=O)=O)c2c(c1)CCO2 64348,c1(CC(C)NCC2CC(CC(=O)O)C2)ccccc1 64349,c1(C(=O)NC2C(C(C)(C)C)N(C(=O)C(=O)N(C)C)CC2)nnn2c1CCCC2 64350,C(N=c1[nH]c2ccc(N)cc2s1)C1CCCCN(C(c2nn(CC)c(C)c2)=O)C1 64351,c1(OC)cc(C)c(C(=O)NC2(CCNC(C34CCCC3C4(F)F)=O)CC2)cn1 64352,c1(OC)c(Br)cc(CN2C(C(=O)NC(c3ccc(I)cc3)C)CC3CC23)cc1Br 64353,C(C(C(C)C)NC(=O)C(C#N)=C1CCCC1)NC(C(C)OCCOC)=O 64354,CC(C)(C(=O)NCC1CCC(NC(=O)CN2CCCC2=O)C1)c1cc[nH]n1 64355,c1(N2C(C(=O)NC(c3cnccn3)C)CNCC2)ncnc2c(F)cccc12 64356,c1(C(N2CCCC(C(C)NC(c3cc(C)sn3)=O)C2)=O)n[nH]c2cc(Cl)ccc12 64357,Cc1cnn(CCC(N2C(C(N3CC(OCCF)C3)=O)CC2C)=O)c1 64358,C1(NC(CCc2cnc(C)o2)=O)CC(C(=O)NC(c2cccnc2F)C)=CC1O 64359,C1(CNC(C2C(=C)C2)=O)CN(C(=O)Cc2ccc(Cl)cn2)CC12CC2 64360,CC1(C)CCN(C(c2csnc2Cl)=O)C1CNC(c1cc(C2CCCC2)no1)=O 64361,c1(C(C)C)cccc(CC(=O)NCCOCCCNC(=O)C(O)C(F)F)c1 64362,C1(NC(c2nc(C)oc2C)=O)CCN(C(=O)C(C)Cc2cnn(C)c2)CC1F 64363,CCC(CC(=O)NCC1CN(C(c2ccoc2C)=O)C2COCC2O1)C(C)(C)C 64364,C(CO)(C(=O)N1CCCC1CN(C(=O)C(C)OC1CCCC1)C)OC 64365,c1(C(N2C(C)C(C)N(C(C3CC=CCC3)=O)CC2)=O)cn2c(n1)C(=O)N(C)CC2 64366,Cn1cnc2c(C(=O)NCc3ccccc3CNC(C34CCC3C4)=O)cccc12 64367,C1(C(=O)NC(C#C)(C)C2CCOC2)CN(C(c2cccs2)=O)CC1C 64368,C12(NC(c3csnn3)=O)CCOC(CNC(C3C=CC=CC=C3)=O)(C1)C2 64369,c1(C(N(CC(O)CNC(=O)COc2ccc(Cl)nc2)C)=O)cc(F)c(F)cc1F 64370,C1(CCNC(C2CCNC2=O)=O)(C(=O)Nc2ccccc2)CCCC1 64371,C1(NC(CCN(C(=O)Cc2cn(C)cn2)CC=C)=O)CCCCC1C 64372,C(=O)(CCC(C(=O)OC)NC(=O)C(N1CCC(F)C(O)C1)c1cn[nH]c1)OC 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64391,c1(C(=O)NCC2(CNC(c3nc(C)oc3C)=O)CC2)cccn2cnnc12 64392,CCC(CC(C)C)C(=O)N1CC2C(CC(=O)NCC3CC3C(C)C)C2C1 64393,C12(C(=O)NCC3CC(F)CN3C(=O)CC34CCCC3C4)CCN(CC1)C2 64394,N1(C(CC(C)(C)CC(F)F)=O)CC2CCN(C(c3nncs3)=O)CCC2C1 64395,N1(C2CC(C(=O)OC)C23CCC3)CC(NC(=O)OC(C)(C)C)CC(C)(C)C1 64396,C(=O)(C1=NOC2(CCC2)C1)Nc1c(C(=O)OCC)ncc(Cl)n1 64397,C1(CNC(CCN(CC=C)C(C2(CC)CCCO2)=O)=O)COCCN1C 64398,c1(NCC(CNC(CC(CCC)C)=O)C(F)(F)F)ncccc1[N+](=O)[O-] 64399,c1(CC)onc(C)c1C(N1CCC(OCCNC(=O)C(C)=CCO)C1)=O 64400,C(=O)(CC(F)(F)CC(=O)OC)NC(CNC(c1c(CC)n(CC)nn1)=O)C1CC1 64401,Cc1ccc(C)n1CC(=O)NCC(C)N(C)C(c1cc(C(F)F)ncn1)=O 64402,CN=c1[nH]nc(CC(=O)NCC2(NC(=O)C(C)Sc3ccc(F)cc3)CCC2)s1 64403,c1(CC)ccc([N+](=O)[O-])cc1OC(F)F.C(Cl)(C(F)(F)F)N1CCC1 64404,c1(N(C)CCF)cc(S(=O)(=O)N2CCCC2CC(C)(C)C)ccc1C#N 64405,C1(NC(c2nc(COCC)sc2)=O)CCN(C(=O)CCSC)CC(C)(C)C1 64406,C(C)(c1cccnc1)=CC(N1CCC(C(C)(C)C)(CNC(CCCC#C)=O)C1)=O 64407,c1(COC)ccnc(C(=O)NC2CC(C)N(C(=O)Cc3csc(NC=O)n3)C2)c1 64408,CN=c1nc(N(C)CCOCC(F)(F)F)[nH]c(=NCc2ccc(Cl)c(F)c2Cl)[nH]1 64409,c1(-c2cc(C(N(CCC3CC(C(=O)OC)C3)CC3CC3)=O)no2)cccc(O)c1 64410,c1(OC)ccc2c(c1)CC(C(=O)NCC(O)CCNC(=O)CC1CCOCC1)O2 64411,C1(NC(=O)CCN2CCC2)CN(C(=O)CC2CCCC2)Cc2ccnn2C1 64412,N1(C(c2cc(CC)nn2C)=O)CC2CCCC2C1C(N1CC(CO)CC(C)C1)=O 64413,C1(CC(N2CC(CNC(C3CCC(c4ccccc4)C3)=O)C2)=O)CCCC(O)C1 64414,c1(C(=O)NCC2(OC)CN(C(C(COC)OC)=O)C2)cnc(O)cc1OC 64415,c1(C(=O)NC(C(=O)NCC(COC)OC)COC)cc(O)ccc1C 64416,c1(CC)cccnc1C(C)NC(C1CN(C)CCO1)C 64417,C1(NC(C(C)=C(CC)C)=O)CN(C(C2(C3CCCCC3)CC2)=O)C2CCCC12 64418,N1(C(COC2(C#C)COC2)=O)CCOCC(C)(CNC(c2ccc(C)nn2)=O)C1 64419,c1(NC(C2(C)CN(C(C(CC)=CCCC)=O)C2)=O)ccc(O)c(CO)c1 64420,N12CCOCC(C1)N2Cc1nc(C)n(C)n1.c1(OCC)cccnc1.C=O 64421,N1(C(COCC=C)=O)CC(NC(=O)C=Cc2ccc(C)s2)CC12CCOC2 64422,C1(NC(CC2(C=C)CC2)=O)CC2CC(C1)N(C(=O)CC1CN3CCC1CC3)C2 64423,c1(C2(C(=O)NCC3(F)CN(C(C4CCCO4)=O)C3)CCCC2)ccc(F)cc1 64424,N1(C(C2CC(C)(C)N(C(C3CCC(O)CC3)=O)CC2)=O)CC2CCC(O)C(O)C12 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64460,Cc1ccc(OCCC(=O)NC(C)CCNC(c2c(C)cnn2C)=O)c(C)c1 64461,c1(-n2cc(NC(C(=O)NC(CCC=C)C(=O)O)=O)nn2)ccc2nonc2c1 64462,c1(-c2cn(CCNC(c3cccc(C(F)(F)F)c3F)=O)nn2)c(F)cccc1Cl 64463,c1(C(=O)OC)c(C2CC2)csc1NC(=O)C(C(C)C)NC(c1ccccc1C)=O 64464,c1(C(N(CC2CCCN(C(CCCOC)=O)C2)CC)=O)cc(Cl)cnc1C 64465,c1(OC)ccc(NC(C2CC3CC3N2C(c2cnc(O)[nH]2)=O)=O)cc1F 64466,c1(C(=O)NC(C(=O)NC(C(C)O)CO)Cn2cncn2)ccccc1F 64467,Cc1ncnc(O)c1C(=O)NC1CCN(C(=O)C(C)Cc2cccnc2)C1(C)C 64468,C1(NC(C2C(C#C)C2)=O)CCCCCN(C(=O)COc2cccc(CC)c2)C1 64469,C1(CNC(CCC2N(C(CCCOCCOC)=O)CCC2)=O)CC12CCOC2 64470,C12(NC(C(C3CCC3)OC)=O)CCC(CN(C(c3cc(C)c(C)nc3C)=O)C1)C2 64471,C=CCC(C(=O)NC(C)CNC(=O)CC(C)O)NC(C)=O 64472,c1(CCC)cnc2c(C(=O)Nc3cc(OCC)ccc3N(C)C)cccn12 64473,n1(C(C)C)cc(C(N2CC(CNC(=O)C(C)(C)C#N)C3(CC3)C2)=O)ccc1=O 64474,C(=O)(C(C)(C)CC(C)(C)C)N1CCC(CC(N2C(C)CCCC2)=O)C1 64475,N1(C(C2C(=O)NCC2)=O)CC(NC(=O)C(C2CC2)C2CC2)CC12CCCCCC2 64476,c1(C(=O)NC(C(C)NC(CCOCC#C)=O)CO)c(Cl)cccc1Br 64477,C(CCC(=O)NCC(F)CNC(c1csnc1C)=O)NC(=O)OCC 64478,C=CC(C)(CC)C(=O)N1CC(OC)C(NC(=O)C(F)(F)c2cscn2)C1 64479,O=C(CS(=O)(=O)N1CCCCC1)NCCC1CCCCN1C(C1CC=CC1)=O 64480,c1(C(=O)NC2CN(C(c3c(OC)nn(C)c3)=O)C3C2C3)cn(C)c(=O)cn1 64481,C(CCC1CCC1)(C(=O)N(CC(O)CO)CCO)SC.N12CC(C1)NC2=O 64482,Cc1cc(O)c(F)cc1C(N1CCOC(c2cn(CC3(O)CCC3)nn2)C1)=O 64483,C1(C)(C(=O)NCC(CC(=O)N(CCNC(C(C)C)=O)C)C)CCC(=O)NC1 64484,c1(C(N(C2CCN(CC3CCOCC3)CC2)CC#C)=O)csc2c1CCCC2 64485,C(=O)(N=c1ccc(Cl)n[nH]1)c1ccc(NC(C(CCC)(C)C)=O)cc1OC 64486,C#CCCCCC(=O)N1CC2CC2C1C(=O)NC1C2CCCCCC12 64487,C1(NC(CC(CCC)C)=O)COC2(C1)CN(C(C1CSCN1C(=O)CC)=O)C2 64488,C1(NC(C=COCC)=O)CN(C(=O)C=CI)CC2(CCOCC2)C1 64489,C1(NC(C(C)C)=O)CN(C(=O)C(F)C2CCC2)C2(CCOCC2)C1 64490,CC1(C)NC(=O)N(CC(N2CC3(CC(NC(=O)C(F)C4CCC4)CO3)C2)=O)C1=O 64491,c1(C(=O)OC)cc2cc(CN(C3(C)COC3)C)ccc2o1 64492,CCC(C)CC(=O)C(=O)N1C(C(N2CCC23CC(CO)C3)=O)CCC12CC2 64493,C1(C)(SC)CC2(CCC2)C1.C1CC(O)C(=O)NCCNC(=O)CN1C1CC1 64494,CCC(C(=O)N1CCCC1C(C)(C)NC(c1ccc[nH]1)=O)N(C)C 64495,N1(CC(=O)NCCC(C)NC(C2CC3(CC3)C2)=O)CCN(C)CC1 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64584,C1(C(N(C2CCCC2)CC#C)=O)COC2(C1)CN(C(=O)C=CC=CCC)C2 64585,C(CC(F)(F)F)N(C(=O)CC(C)NC(NOCCC#CC)=O)C1CCCC1 64586,C1(N(C(c2ccc(CC)s2)=O)CC)CCCN(C(=O)CCc2ccccn2)C1 64587,N1(C(C(C)=CC2CC2)=O)CCC2(CC1)CCN(C(c1c(C)cc(Cl)cc1N)=O)C2 64588,c1(C(C)=O)cc(C(N2CCOC(C)(CNC(C34CCC3C4)=O)C2)=O)c(C)nc1C 64589,C(c1ccc(Cl)s1)=CC(=O)NC(CNC(C=CCN(C)CC)=O)(C)CO 64590,c1(SCCN(C(c2ccc[n+]([O-])c2)=O)CC)cccc2c[nH]nc12 64591,C1(NC(c2nc[nH]c3nccc2-3)=O)COC2CN(C(C3C4CCOCC34)=O)CC12 64592,c1(OC)ccccc1C(C)(C)C(=O)NCC1C=CCN1C(c1cc(Cl)c[nH]1)=O 64593,CN1CCC(=CC(N2CC(NC(c3ncccc3C(F)(F)F)=O)C(O)C2)=O)CC1 64594,CC1(C)CC(C(=O)N2CCCC2C2(NC(c3ccc(C(=O)O)nn3)=O)CC2)=NO1 64595,c1(N2CC(N(C)C)C(C)(C)C2)nc2c(c(=NCC#CC3CC3)[nH]1)CCC2 64596,C1(c2nnnn2CCCSCC)(NC(CCCC=C)C)CC2(CCCC2)C1 64597,Cc1nc(CNC(C23CC(NC(=O)CSC(F)(F)F)(C2)C3)=O)[nH]c1C 64598,Cc1cc(Cl)cc(C)c1OCC(=O)NCCN(C(=O)COC1CCCCC1)C 64599,CCS(=O)CC(=O)N(C)CCN1CCN(C(C2CCC(=O)C2)=O)CC1 64600,N1(CC(COC)O)CCN(C(=O)OC(C)(C)C)CC1.C1CCC(C)N1 64601,c1(CC)noc(CCCC(=O)NCCN(C(=O)CC#N)CC)n1 64602,CC1(C=CC(=O)NCC2CN(C(C3(CO)CCCO3)=O)CC2(F)F)CCOCC1 64603,CCCC(C(=O)NC(c1cn(CCOCCOCCO)nn1)(C)C)S(N)(=O)=O 64604,C(=O)(C(C1CC1)N(C(=O)CC1CCOC1)C)NCC(C1CCCC1)C 64605,N1(C(c2c(Cl)cn(CCC)n2)=O)CCCN(C(=O)CCN(C)C(C)C)CC1CO 64606,C(C1=CCN(C(=O)CN2CCC(O)CC2)CC1)NC(C(C(C)C)NC(C)=O)=O 64607,N1(C(C(CC)C)=O)CCCC(C)(NC(=O)CCc2cccnc2Cl)C1 64608,N1(Cc2c(CC(=O)OC(C)=O)cccc2)CCc2cc(NC(C)=O)ccc2C1 64609,C(=O)(CC(O)C(Cl)(Cl)Cl)NCCC(C)NC(CC(C(=C)C)O)=O 64610,C1(C)(CC)CCCC1NC(=O)C(C1CN(C(C2CC3(CSC3)C2)=O)C1)OC 64611,C1(C(N2CCC3C(CCN3Cc3nccnc3Cl)C2)=O)CCCC2CCCCC12 64612,c1(N(C)C)ccc(C=CC(=O)NC2CC(O)CN(C(c3ccc(F)o3)=O)C2)cc1 64613,CON1CCC(CN(CCF)C(c2nc(C)n(-c3ccccc3Cl)n2)=O)CC1 64614,c1(C(N2CCC(C)(NC(=O)Cc3ccns3)C2)=O)cnn2ccc(O)nc12 64615,C(=O)(C(C(C)C)C1CCC1)N1CC(C(=O)NCCCOC)(CC)C1 64616,C1(C(=O)NC(C(C)NC(c2c(C)nn[nH]2)=O)CO)CN2CCCC1C2 64617,C1(NC(=O)OC(C)(C)C)CC(S(C)(=O)=NC(=O)C23CCC(CC2)OC3)C1 64618,CC1=C(C(=O)N2CC(NC(C3(O)CCCC3)=O)CC23CCC3)C(=O)OC1(C)C 64619,c1(C(N2CCC(N(C(C(CC)N(C(N)=O)CC)=O)C)C2)=O)cc(C#N)[nH]c1C 64620,C(=O)(C1=CC2C=CC(C1)C2)N1CC(NC(c2n(C(C)C)ccn2)=O)C(N=[N+]=[N-])C1 64621,C12(NC(C(C)=C(C)C)=O)CCC1CN(C(=O)Cc1sc(C)nc1C)C2 64622,C(=O)(C(C)(C)C1=CCSCC1)NCC1N(C)CCN(C(c2csc(O)n2)=O)C1 64623,c1(C(=O)NCC2CCC(NC(c3c(SC)cnn3C)=O)C2)cc(C)c(O)c(N)c1 64624,Cc1nc2ncccn2c1C(N1CCC(C(=O)Nc2nccs2)CC1)=O 64625,c1(CC)cnoc1C(=O)N(CCC(C)NC(=O)Cc1cscc1Br)C 64626,c1(NC(N)=O)ccc(C(=O)NCC2CCN(C(C3CCSC3)=O)C2)cc1 64627,c1(OC)cccc(CC(=O)NC(C2COCCN2C(c2cnco2)=O)C)c1 64628,N1(C(CNC(C)=O)=O)CC2CC(NC(C3(C)C=CCCC3)c3ccsc3)C2C1 64629,N1(C(C(CC)NC(C2CCC(=O)N(C)C2)=O)=O)CCC12CCC(C)CC2 64630,C(=O)(CC(C)(O)C(F)(F)F)NCCC(C)(C)NC(c1c(C)n(CC(C)C)nc1)=O 64631,N1(C(COC)=O)CCC2(NC(c3ncn4c3CCC4)=O)CCCCCC12 64632,N1(CC(=O)NC2CCC2)CCN(Cc2cccc(Br)c2)CC1 64633,C1(CCOC)(NC(=O)C(C)c2cccs2)CCN(C(C2CC2(Cl)C(=O)OC)=O)C1 64634,C1(NC(CCN(CC)CC)=O)CN(C(c2cc(CO)[nH]n2)=O)C2CCCC12 64635,CC1CC(C(N2CCCN(C(=O)CCC(F)F)CC2)=O)C1C1CC1 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64654,CC1CCC(NC(=O)CCOc2ccc(C(N)=O)cc2)CN1C(c1cc[nH]c1)=O 64655,c1(CNC2CC(C(=O)Nc3ncc(C(=O)OC)nc3)C2)c[nH]c2ncc(C)cc12 64656,C(=O)(CC(F)(F)F)NCC1(O)CC(NC(CCc2onc(C)n2)=O)C1 64657,C(=O)(CS(C)(=O)=O)NCC(C)(F)CNC(=O)C(C)(C)n1ccnn1 64658,CC(CCCNC(=O)COCC1(Cl)CC1(F)F)NC(=O)C=CSc1ccccc1 64659,c1(C(C)OC)nc(-c2ccnc(C)c2)n(-c2cccc(C(N)=O)c2)n1 64660,C1(C(=O)NCC(C2CC2)N(C(=O)CCOCC2CC2)C)(OCC)CCCCC1 64661,N(C1c2sccc2OC(C)(C)C1O)C(C(C(C)C)OCC(C)C)=O 64662,c1(C(C)Oc2ccc(NC(C)C(C)(C)CN(C)C)cc2)cc(F)cc(S(N)(=O)=O)c1 64663,c1(C(CNC(C2CC(C)(F)C2)=O)NC(=O)Cc2sccc2Cl)ccc(F)cc1 64664,N#Cc1ccc(C(=O)NC2COCC2NC(=O)CCc2ccncc2)cc1F 64665,c1(C(=O)NCC2CCN2C(c2cn(C3CC3)cn2)=O)c(F)cncc1Cl 64666,C1(=CC(N2C(C(C)NC(Cc3cnc(C)[nH]3)=O)CCC2)=O)CCCCC1(C)C 64667,C1(CC(=O)N(CC(N2CC(N(C)C3CC3)C2)=O)C(C)C)CCC(C)C(C)C1 64668,C1(N(C(=O)CC(C)C2CC2)CC#C)CCN(C(C2CC(OC)C2)=O)CC1 64669,CCC(C)CC(C)C(=O)N1CC(CO)C2(C1)CN(C(c1cnn(C(F)F)c1)=O)C2 64670,N1(C(C2(CF)CCOCC2)=O)CCOC2(CCN(C(C34COCC3C4)=O)CC2)C1 64671,C1(C(N2C(CNC(C3C4CC5C(C4)C35)=O)CCC2)=O)CC2CCC(C1)C2=O 64672,N1(C(C=C(C)Cl)=O)CCN(CCNC(c2nn(C)nc2Br)=O)CC1 64673,c1(C(C(=O)NC)N(C)Cc2cccnc2OC)ccc(C(F)(F)C(F)(F)F)cc1 64674,c1(CN2CC(C(=O)Nc3c(OC)ccc(Cl)c3)OCC2)cc2ccoc2cn1 64675,c1(NC(CC2C(NC(COC(CC)C)=O)CC2O)=O)ccc2c(c1)CCO2 64676,c1(C(=O)NC(CNC(=O)CCn2ccnc2)C2CCC2)cc(F)cc2nn[nH]c12 64677,n1(CC(N2CCN(C(CCCC=C)=O)CC2C(F)F)=O)ccc(=O)c([N+](=O)[O-])c1 64678,N1(C(C(=O)NC2CC(F)(CNC(C(C)n3ccnc3)=O)C2)C)CCC(O)CC1 64679,C1(NC(c2n(CC)nnc2)=O)(CF)CCN(C(=O)CN2CC3C=CC2C3)C1 64680,c1(C(=O)NCC(CNC(C2NC(=O)OC2)=O)C(F)(F)F)cnc2c(c1)CCCO2 64681,C12(C(N(CC(N3CCC3CC)=O)CCC)=O)CCCCC1C2 64682,c1(NCc2c(C)ccs2)ncccc1S(=O)(=O)NCc1c[nH]c(=N)s1 64683,C1(OC)CC(C(=O)NCC(O)CC2CCCC2)N(C(=O)CNC=O)C1 64684,CC1=CCC(C(N2CC(C(=O)Nc3cc(C)nn3-c3ccccc3)C2)=O)CC1 64685,CCC(CN(C)C)CC(=O)NC1(CNC(C2CC23CCC3)=O)CCC1 64686,C(CCCCC)=C(C(=O)N(C(C=CC(=O)OC)C)C(=O)C=Cc1ccsc1)F 64687,N1(C(c2ccc(C)s2)=O)CC2(CCOCC2)CC1CNC(=O)CC(C)C 64688,CCC(C)CCCC(=O)N1CC2C(NC(=O)CNC(c3ccc(F)cc3)=O)C2C1 64689,C(=O)(C(C)CC(C)(F)F)NC(CCNC(C1(OC)CS(=O)(=O)C1)=O)C 64690,C1(N(CCOC)C(c2cn(C)nn2)=O)CCN(C(=O)C(c2cnccn2)C)CC1 64691,C1(C(=O)NC2(C)CCN(C(c3cnc(C)n3C)=O)C2)CCCC2(CCC2)O1 64692,C(=O)(C(O)C(C(C)C)OC)N1CC(OCCC(N2CC(CC)(OC)C2)=O)C1 64693,C(CO)(CCCCNC(c1cc[n+]([O-])cc1)=O)NC(c1c(CC=C)cccc1)=O 64694,C1(CCC#C)CCCN(C(=O)C(C2CN(C(=O)C(C)OCCCC)C2)OC)C1 64695,C(=O)(C1=C(C)C(C)(C)OC1=O)NCC(C(=O)OCC)(C)CC 64696,c1(OC)cnc(C(=O)NC2CCC(NC(=O)CC3CCC(C)(C)C3)C2)cn1 64697,c1(C(CF)NC(=O)NC2(CCCCO)CCOC2)ccc(Cl)cc1Cl 64698,C(C(C)C(=O)NCC1(NC(c2ccn(CCF)n2)=O)CCCC1)OC 64699,N1(C(C(CSC)O)=O)CCC(C)(CNC(c2ccc(C)n2C)=O)C1 64700,C1(NC(c2c(CC)scc2)=O)COC2(CNC(C3COCCC3(F)F)=O)CC1C2 64701,C(=O)(C(C(C)CC)N(C)C(c1coc(COC)n1)=O)N(CC=C)CC1CC1 64702,c1(C(N2CC=CC(NC(C(CC)(C)COC)=O)C2)=O)sc2ncccc2c1N 64703,CCC(CNC(=O)C=NOC)(CC)C(=O)NC1CCNC(=O)CC1 64704,CC1(C)CC(C(=O)NCC23CC(CN2C(=O)C=Cc2cnc[nH]2)C3)CNC1=O 64705,N1(C(C2(CC)CC2)=O)CC2(C1)CN(C(=O)Cc1nc(C3CC3)oc1C)CC2CO 64706,CC1CCCC=C1C(=O)NCCC1CCN(C(=O)CN(CC(C)(C)C)C)CC1 64707,c1(C(=O)NC(C)(CNC(C2(C(F)F)CC2)=O)C2CCC2)csc(O)n1 64708,c1(CCCC(=O)NCC(CC)NC(=O)C=Cc2cnn(C)c2)cccc(Cl)c1 64709,C1(NC(COCCCC)=O)CCC12CCN(C(=O)C(=O)Nc1cccc(C)c1)CC2 64710,c1(N2CCC(CC=C)(NC(=O)C(COC)OC)CC2)cnc2ccccc2n1 64711,c1(N2CC(C3N(C(C4CCCN4C4CC4)=O)CCCC3)C2)cccc(F)c1[N+](=O)[O-] 64712,CC1OCCN(C(C2CN(C(C3(O)CCSC3)=O)CC2(C)C)=O)C1CO 64713,O=C(CCc1cccc(OCC(F)(F)F)c1)N=c1[nH]n(C2CC2)c2ccccc12 64714,C#CC1(O)CC(C(N2CCCC2CN(C(=O)C(c2ccncc2C)C)C)=O)C1 64715,C(=O)(C1=C(Cl)CCCC1)N1CC(C)CC(C(N(C)Cc2nc(C)on2)=O)C1 64716,C1(C(N2C(C)CN(C(=O)CCc3cccs3)CC2)=O)CCN2CCOCC12 64717,C(=O)(CC(C(C)C)OCC)NC1(C)CN(C(c2cc(CCC)c(C)s2)=O)C1 64718,CC(C(=O)N1CCN(C)C(C(=O)NCCCN(CCO)CCO)C1)C(F)(F)F 64719,c1(C(=O)NC(C2CCCN2C(=O)CNC(N)=O)C)cc2ccc(Cl)c(F)c2[nH]1 64720,C(C(=O)NC(C)C(CO)NC(C1CCN(C(=O)CC)C1)=O)(C(C)C)NC(C)=O 64721,C1(C)(NC(C2C(C)CCC2)=O)CCN(C(C2(c3ccccc3Br)CC2)=O)CC1 64722,C(C)(CO)(C(=O)N1CCC(OCCNC(=O)CNC=O)C1)OC 64723,C1(NC(=O)C(c2ccccc2)O)CC2CC1CN(C(C1(F)CCCC1)=O)C2 64724,C1(C)(CNC(CCNC(COC)=O)=O)CN(C(c2ccnc(C3CC3)n2)=O)CC1C 64725,n1(CC(=O)N(C2CCN(C(c3cc(C)no3)=O)CC2C)C)ccc(=O)n(C)c1=O 64726,c1(CCC(=O)NC(CC)(C)CNC(C2(CF)CC2(F)F)=O)cccc(Cl)c1 64727,C1(NC(C(CSC)OC)=O)CCN(C(c2cc(-c3ccco3)on2)=O)C12CCC2 64728,N1(C(c2c(CNC(C3CC(=O)NCC3)=O)cc[nH]2)=O)CC2COCC(C2)C1 64729,Cc1c(C(=O)NC(C2(C(=O)O)CCOCC2)(F)F)noc1-c1ccccc1 64730,NS(=O)(=O)CCCCCCC(=O)NCCCOc1ccccc1F 64731,c1(C(N2C(C(=O)NC3CC(F)(F)C3)CSC2)=O)ccncc1Cl 64732,N1(C(Cc2ccc(CC)cc2)=O)CCN(C(=O)Cn2cc(C)cn2)C(C2CC2)C1 64733,c1(C(N(C2CC(NC(C3ON=C(CC)C3)=O)C2)C)=O)cc2c(Cl)cccc2s1 64734,Cc1scc(C(=O)N(CCC(=O)NC(C(O)CO)C2CC2)C2CC2)c1C 64735,S(=O)(=O)(c1cccc(N2CCOCC(O)C2)n1)N(CC)CC 64736,N1(C(CCCOCC)=O)CCN(Cc2cn(CCOC3CCOC3)nn2)CC1 64737,Cc1n[nH]c(C)c1CC(=O)N(CC(O)CNC(=O)C(C)Sc1ccccc1)C 64738,C1(NC(CC(C)(C)NC(Cc2ccc(C)s2)=O)=O)C(O)C2CCOC12 64739,C12(C(=O)NC(CCOC)C)COC(C1)C(NC(=O)C=CC1CCCCC1)C2 64740,C1(CC(N2CC(C)CC(C)C2)=O)CCC2(CC1)CCN(C(=O)COCCO)CC2 64741,CCC(C)C(O)C(C)C(=O)NCC1CN(C(=O)CNC(=O)CC)C2CCN1C2 64742,c1(C(=O)NCC2N(C(c3cn(C)nn3)=O)CCC2)c(O)cccc1O 64743,N1(C(C(C=C)O)=O)CC(O)CC1CNC(=O)CNC(=O)NCC1CCCC1 64744,CC1CC(c2nc(-c3cc[nH]n3)nn2-c2ccc(C34CC(C3)C4)cc2)=NO1 64745,N1(C(C(=Cc2cccs2)C)=O)C2CCCC1CN(C(=O)C(c1cccnc1)O)C2 64746,c1(C(N(C)CCOCCN(C)C(C2(Cl)CC2(F)F)=O)=O)cccn2[nH]c(=N)nc12 64747,c1(C(=O)NCCC(C(C)C)NC(C=CSC)=O)cc2cccc(F)c2o1 64748,CC1CCC(CN2CC(N3CC(C(=O)NN4CCCC4)CC3=O)C2)NC1 64749,N1(C(=O)CCC2CC2)CCCCC1C1CCCN(CC2(O)CCC2)C1 64750,c1(C(C)NS(c2ccc(NC(=O)OCCC)s2)(=O)=O)sc2ccccc2c1C 64751,CCC(C)(CCC(C)C)C(=O)NC1CC(CCNC(c2c(Cl)ccnc2C)=O)C1 64752,c1(OCC(=O)NC(C)C(C)NC(c2ccc(N)c(N)c2)=O)ccc(F)c(F)c1 64753,N1(C(c2ccc(CNC(c3cc(OC)n[nH]3)=O)cn2)=O)CCC2C(C(N)=O)C2C1 64754,CC1(C)CCCC(C(=O)NCC2CC(NC(=O)C(c3ccccc3)O)C2)O1 64755,CC(CCC(C)(C)C)C(=O)NC1CN(C(=O)CN2CSCC2=O)CCC1O 64756,c1(OCCOC)ccc(-c2nc(CC(C)C)nn2C(C)C(F)(F)F)cc1 64757,c1(CN2CC(C)(NC(=O)Nc3ccc(SC)cc3)C2)ccc(CO)c([N+](=O)[O-])c1 64758,N1(C(C2COCCO2)=O)CCC2(CCCN(CC=Cc3ccccc3)C2)C1 64759,c1(COC)nc(C)c(C(=O)NCCCN(C(=O)Cc2csc(Cl)c2)CCO)s1 64760,N1(C(C2(CN(C)C)CC2)=O)CCOC2(C1)CN(C(c1ccnnc1O)=O)C2 64761,CC1CC(CNC(C2(F)CCOC2)=O)CCN1C(C1CC(=O)C1)=O 64762,Cc1cnc2c(cnn2CC(=O)NC2CCCN(C(c3cccs3)=O)CC2)c1 64763,c1(CC(=O)N(CC(C(C)C)NC(C(c2ccccc2)OC)=O)CCO)cc(C)cc(F)c1 64764,c1(NC(=O)NC(CC)CNC(C2CC2C(=O)OC)=O)ccccc1C(F)(F)F 64765,c1(CCNC(N2CCC(CNC(CC)=O)C2)=O)ccc2c(c1)COC2 64766,C(c1cc(C)cc(C)c1)=CC(=O)NCCN(C(C(C(C=C)C)C)=O)CC 64767,C1(NC(c2c(C)ocn2)=O)C2CC3C1C3C2C(N1CC(OC(=N)O)C1)=O 64768,CCC(C)(CO)C(=O)N1CCCC(N(CCO)C(c2ccc(C(F)F)c(N)c2)=O)C1 64769,C(CN=c1ccnc(N(C)Cc2cccc3ccccc23)[nH]1)C1C(C)C1 64770,c1(C(=O)NCC2C(NC(c3ncc(OC)nc3)=O)COC2)cc(C)ccc1Cl 64771,CC1(C)CC(NC(C2C(O)CCN2C(=O)CC#N)=O)C12CCC2 64772,Cc1ccc(CCC(=O)NCC2CCC2NC(=O)CCC(=O)N(C)C)cn1 64773,c1(C(N(C(CCNC(C(CC=C)OC)=O)C)C)=O)ccc([N+](=O)[O-])cc1 64774,C(=O)(C1=NOCC1)N(C(CCNC(C1CC(CC)C1)=O)C)C 64775,N1(C(C2CC=CCC2)=O)CC2=C(C1)CN(C(C1(O)CC(F)(F)C1)=O)C2 64776,Cc1cc(C2CCC2)ncc1C(N1CCC(NC(C2CCC(C)(C)O2)=O)C1C)=O 64777,N1(C(COCCCC)=O)CC(NC(=O)C(C)(C)CF)C(SC)C1 64778,c1(CC(N2CC(C)C(NC(c3ccn(CCF)n3)=O)C2)=O)nc2ccccc2s1 64779,C#CC(C)(C)C(=O)NC1CNCCC1c1ccc(OCC)cc1 64780,c1(C(=O)NCC2(O)CC(NC(C(C)OC)=O)C2)cc2c(nc1O)CCCC2 64781,c1(CC)[nH]c(C(=O)NC(C)(CNC(C2CCOC2)=O)c2cccs2)nc1Cl 64782,O=C1CC(C(=O)NCCC2COCCO2)N(C(=O)CC(Cl)Cl)C1 64783,CCCCCCCN(C(=O)C(C1CCCO1)NC(=O)C=CC1CCC1)C 64784,C1(NC(C2CCC(C(C)C)CC2)=O)CN(C(C2CC2(C)Br)=O)Cc2nccn2C1 64785,Cc1ccccc1C=CC(N1CC(C(C)NC(c2cccc(F)n2)=O)C1)=O 64786,C(CN=C(NCc1ccc(C2CC2)c(F)c1)N1CCC(C)C1C)OC 64787,C1(C(=O)NCCC(C)CCNC(c2cscc2Cl)=O)CCc2cn(C)nc2C1 64788,C(=O)(CCCCC(N)=O)N1C(c2cn(-c3c(F)ccc(OC)c3)nn2)CCC1 64789,N1(C(C(C)C)=O)CCC(C2CCN(C(=O)C(F)C3CCC3)CC2)C1 64790,c1(C(N2CCNC(C(N3CCC(O)C(O)C3)=O)C2)=O)cc(I)ccc1F 64791,Cc1[nH]nc2c(C(N3CCC3CNC(c3ccc4cncn4c3)=O)=O)cccc12 64792,c1(C(N2CC(OC)C(NC(=O)CC3(C)CCCO3)C2)=O)cn2ccccc2n1 64793,C(CCCC(C)(C)NC(=O)CCCN(C)C)NC(CSCC=C)=O 64794,C(=O)(CCCCCC(C)C)NCCCN(C(C=Cc1c(C)noc1C)=O)C1CC1 64795,C(=O)(C1c2ccccc2C2CC1C2)NCC1CCC(C)C1 64796,C1(C(COC(C(C)Cn2cccn2)=O)=O)CCN(C)C1=O 64797,CC1(C)CN(C(C2CCN(CCO)C(=O)C2)=O)CC1NC(=O)CCc1nc[nH]n1 64798,N1(C(C(CSC)C)=O)CC(CNC(C2(C)CCC3CC3C2)=O)CC1(C)C 64799,c1(C(N2C(C)(C(N3CCN(C)CC3)=O)CC2)=O)cc(Cl)cc([N+](=O)[O-])c1 64800,Cc1cc(CN2CC3CC3(C(=O)Nc3cc(C(F)(F)F)c(Br)cn3)C2)ccc1Br 64801,c1(C(N(CCCCNC(CC2CCC(C)C2)=O)C)=O)cccc(F)c1Cl 64802,C1(NC(=O)C2=CCN(C(c3ccc(CO)s3)=O)C2)CC2CCCC(C1)C2 64803,CC1CC2CC(C(=O)N(C3CN(C(=O)CCn4cccn4)C3)C)(C2)O1 64804,c1(OC)cncc(NC(=O)C(C2CCC2)NC(=O)C(O)CCN(C)C)c1 64805,c1(CCC)c(C(=O)NCC2CC2CNC(=O)C=Cc2cccnc2)nnn1CC 64806,Cc1cccc(C(=O)NCCCCCNC(=O)C(c2cnn(C)c2)O)c1O 64807,N1(C(C(CC=C)CC)=O)CCCCCC(NC(c2onc(C)c2C)=O)C1 64808,Cc1ccc(C)n1CC(N1CC(O)(C(C)NC(c2cnn(C3CC3C)c2)=O)C1)=O 64809,Cc1cc(=NC(CF)c2ccccc2Cl)[nH]c(C2(C(=O)OC(C)(C)C)CC2)n1 64810,C1(CNC(C2C(OCC)CCC2)=O)(OC)CCN(C(=O)C(C)NC(C)=O)C1 64811,c1(C(=O)NC(CC#C)(C)C(=O)NCCCN=[N+]=[N-])ccc2cc[nH]c2n1 64812,N1(C(CN(C)S(N)(=O)=O)=O)C2CCC1CC(F)(CNC(=O)CC(=O)N1CC1)C2 64813,Cc1cc(C)[nH]c(=NCc2cn3ccc(-c4ccnc(OC(C)C)c4)cc3n2)n1 64814,N1(C(C(C(=C)C)(C)O)=O)CC(NC(c2ccc(CC3CC3)s2)=O)C(C2CC2)C1 64815,Cc1cc(=O)n(C)nc1C(N1CCCCC1CN(C(=O)C(C)(Cl)Cl)C)=O 64816,C1(c2cn(CCCC)nn2)CCN(C(=O)C=CC(C)C)C(C)C1.Cc1sccc1N 64817,Cc1cc(Br)cc(C)c1C(=O)NC1CN(C(c2c(O)cncc2F)=O)C1 64818,Cc1ccc(O)c(NC(=O)CCC(C)(C)NC(C2CCCCO2)=O)c1 64819,C1(CC=C)(NC(=O)CCc2ccsc2)CCN(C(=O)COCCCF)C1 64820,N1(C(=O)OC(C)(C)C)CCC(CN2CCC23CCCC3)CC1NC(=O)C(F)(F)F 64821,C1(CNC(C23CC(C(=O)OC)(C2)C3)=O)(NC(=O)CC2CSCCS2)CCOCC1 64822,N1(C(C(CCS(C)=O)O)=O)CCN(C(c2cnns2)=O)C2(CCC2)C1 64823,C(CCCCC(=O)NC1CC(CNC(=O)CC2OCCOC2(C)C)C1)NC(C)=O 64824,C1(OCC)CC(Nc2nc(OCC)ccc2N(C)C)C12CCCC2 64825,CCCC(C)CC(=O)NC1CC(F)(CNC(c2cc(C)nn2C(F)F)=O)C1 64826,N1(C(c2cc(C(C)C)[nH]n2)=O)CC(NC(c2c(Br)cnn2C)=O)CC(C)C1 64827,Cc1cc(O)nc(C)c1C(=O)NCC(c1ccccc1)CNC(C)=O 64828,c1(CNc2c(CC(=O)NCc3ccc(F)cc3)cccc2)cnc(Cl)cc1F 64829,CC#CCC(C(=O)NC(c1cn(C)nc1C)C)NC(c1cn(C(C)C)nn1)=O 64830,C1(NC(=O)CC2CC3(CC3)C2)CCN(C(=O)CS(=O)(=O)Cc2cccs2)CC1F 64831,C(CC(C(=O)NCc1ccc(F)cc1)NC(C1C2CCC(F)C12)=O)SC 64832,C1(CC(=O)N(C2C(C)CCC2)C)CCCN(C(C2(C)CCCCCC2)=O)CC1 64833,Cc1ccc(CCN=C(NCC(C)(C)C2CC2)NC(C)C2CC2)c(O)c1.C1CC1 64834,c1(C(=O)NC(C2(O)CN(C(c3c(SC)cn(C)n3)=O)C2)C)nc2sccn2c1C 64835,c1(C(=O)NC2COCCN(C(C(C)(Cl)Cl)=O)C2)cccc2cnsc12 64836,N1(C(Cc2nc(C)sc2)=O)CC(O)CC1C(=O)NCCOCCN(C)C 64837,Cc1ccc(CN(C(=O)CNC(=O)C(C(C)C)NC(c2ccco2)=O)C)c(C)c1 64838,Cn1ncc2c1CN(C(C1CC3CC3N1Cc1cc(F)cnc1Cl)=O)C2 64839,C1(C(=O)NC(C2CC(NC(=O)CC3CCCO3)C2)C)CC(C(=O)OC(C)(C)C)C1 64840,C1(C(=O)NC(c2ccc(F)cc2)CC)CC(O)CCN1C(c1sc(C)cc1C)=O 64841,C1(C(=O)NC(CCC(C)C)C)CC1C1CN(C(C2(O)CCCC2)=O)C1 64842,CCC(C(=O)N(C1CCN(C(c2ccsn2)=O)C1)CCO)SC 64843,c1(C(=O)Nc2ccsc2)ccc2nc(-c3ccc(O)nc3)cn2c1 64844,c1(C(N2C(C(C)(C)C(=O)NCc3ccccc3)CCC2)=O)cc2ncccc2[nH]1 64845,C1(C(N(C[Si](C)(C)C)C(C)(C)C)=O)CCCN(S(N)(=O)=O)C1 64846,CC1=C(C(=O)N(C2CCN(C(=O)CCC3CC(F)(F)C3)C2)C)CCO1 64847,N1(C(C=C(CC)CC)=O)CCC2CN(C(c3c(N)sc(C)c3C)=O)CCC2C1 64848,N1(C(C2CCCCC2C(F)(F)F)=O)CCC2(CCNC2=O)C1 64849,c1(CC(N2CCC(N(C)C(c3ccnc(C(F)F)c3)=O)C2)=O)cc(F)ccc1F 64850,N1(C(C(=Cc2ccccc2)C)=O)CCC2(CC2NC(=O)CC23CCCC2C3)C1 64851,c1(C(=O)Nc2cccc(C(=O)O)c2F)noc2c1CCc1sccc1-2 64852,c1(C(=O)NC(COCCCNC(c2ccc(C)nc2)=O)(C)C)nccc(F)c1Cl 64853,C=C(F)C1(CC(N2CCCCC2CC(=O)NCC#CC2CC2)=O)CCC1 64854,Cc1ncsc1C(=O)NC1CCC(NC(=O)CO)C1.C(CC=O)OCCNC(N)=O 64855,N1(Cc2c(CC)noc2)CCCC(NC(c2cc(C(F)F)nn2C)=O)C1C 64856,C(=O)(C(C)(C)C(=O)NCc1occc1C(N1CCSC2CCC12)=O)N(C)C 64857,c1(CC)sc(C(=O)NC(C2(O)CN(C(c3cccn3C)=O)C2)C)cc1Br 64858,c1(OCC=C)ccc([N+](=O)[O-])c(C(=O)NC2CCCCN(C(=O)C=CCC)C2)c1 64859,C1(C(=O)NCC2(C(N)=O)CN(C(c3cc(C(C)C)on3)=O)C2)CCCC(F)C1 64860,CC(CC(=O)N1CC(F)(CF)C1)C(C)(C)NC(=O)C(c1ccccc1)F 64861,C1(CN(C(C=C(C)C(C)(C)C)=O)C)CC(F)CN1C(=O)COCC(F)F 64862,C1(C(N(CC(=O)NC(c2ccccc2O)C)C2CCC2)=O)CC1C1CCC1 64863,c1(C(c2ccccc2OC)C(=O)OCC)ccc(C)cc1CC.C1(=O)CN1 64864,C1(CNC(C=Cc2ccc(CC)o2)=O)CC(F)(F)CN1C(=O)CC1CNC(=O)C1 64865,N1(C(CCCC(OC)OC)=O)CCCC12CCN(C(=O)C(CO)c1ccccc1)C2 64866,C(CC(=O)NC(C)(C)CCNC(=O)COc1ccc(Cl)c(F)c1)(C(F)(F)F)OC 64867,CCC(C)(C)C(=O)NCCN(C(=O)CCc1nc(O)n[nH]1)CC(C)O 64868,C(c1ccccc1Cl)=CC(=O)NC(CNC(C1CCOC1)=O)CC(F)(F)F 64869,C1(C(N(CCN(C(=O)Cc2cn[nH]c2)CC)CC)=O)(OC)CCC(C)C1 64870,N1(C(C2(C)CC(C)C2)=O)CC(NC(c2c(C3CCC3)cnn2C)=O)CC2(CC2)C1 64871,c1(OC)n[nH]cc1C(=O)NCC(CNC(=O)Cc1ccsn1)CO 64872,c1(C(=O)NCCNC(C(C)C)=O)csc(C(C)NC(=O)C(=O)NC2CC2)c1 64873,c1(C(=O)NC(C(C)NC(c2cc(OC)ns2)=O)C)cccc(C(C)(F)F)n1 64874,N1(C(C2C(NC(CCOC(C)=O)=O)CCOC2)=O)CC2(CNC(=O)N2)C1 64875,N1(C(COC2CCN(C(C3(OC)CCC(C)C3)=O)C2)=O)CC2CCC(C1)C(=O)N2 64876,C1(C)(c2cn(Cc3cc(C)on3)nn2)CCCN1C(=O)C(c1ccc(Cl)s1)C 64877,C1(NC(C2CCC(NC(C)=O)CC2)=O)CCN(C(C2CCCC(=O)N2)=O)C(C)C1 64878,N1(C(c2c(C)n(C3CC3)nc2)=O)CCN(C(c2coc(C#N)c2)=O)CC1CF 64879,C(=O)(C(O)CC[S+](C)C)NCC1CC(OC)CN1C(c1cccc(Cl)c1O)=O 64880,N1(C(C2C(C=C)C2)=O)CCc2c(CNC(=O)CCCc3nccs3)cccc2C1 64881,CON(CC1CCCC(C)C1)S(=O)(=O)c1ccc(F)c(F)c1F 64882,C1(CNC(C(=O)N(C2CC(C(N)=O)C2)C)=O)(CO)CC2CC2C1 64883,C(=O)(C(C)(F)C(C)(C)F)N1CCC(CNC(C(C(=C)C)(C)C)=O)CC1C 64884,C1(NC(CCN(C)CCO)=O)CCCCCC1C(=O)NCC1CCSC1 64885,Cc1ccc(-c2ccc(CN(CC(O)CO)C)cc2)cc1F 64886,C1(CN(C(C2CC(O)(CC#C)C2)=O)C)CCCCN1C(C1CCOC1C)=O 64887,c1(C(N(CCCCNC(CC2C(OC)CC2)=O)C)=O)cnn(CCC#N)c1C 64888,c1(-n2c(C)nnc2)ccc(C(=O)NC2CN(C(C3CCN(C)CC3)=O)CC2O)cc1 64889,C1(N(C(C(C)SC)=O)C)CCC(CNC(=O)Cc2sccc2Cl)CC1 64890,n1(CCSCC=C)c(N2CCCC(OC)C2)nnc1C(c1ccc(C)cc1)O 64891,c1(CCNC(=O)NC2C(CN(C)C)CCC2)nccc(=O)n1C 64892,CC1CC=C(C(=O)N2CCC(F)(F)C(CNC(C3CCCO3)=O)C2)CC1 64893,N1(CC(N2C(C(=O)O)CCC(F)C2)=O)C(=O)C(=O)N(Cc2ccccc2)C1=O 64894,CC1(C)CC(C)(CN2CC(C(=O)O)CC23CCC3)CN1 64895,Cc1cn(C)c(C(c2nnnn2C2CCCC2)NCCCCCCN(C)C)n1 64896,C1(c2nccn2C)CCN(C(C=CSC)=O)CC1 64897,N1(C(C)C(=O)N(C)CCNC(C2CC(CSC)C2)=O)C(=O)C2CCCCC2C1=O 64898,N1(C(CCOCCC)=O)CC(NC(c2[nH]nnc2CC)=O)CC1(C)COC 64899,Cn1cc(Cl)c(C(=O)NCCc2ocnc2CNC(=O)CC2CC3CC3C2)n1 64900,c1(CN(C(=O)C(=O)N(C)CC2(O)CCC2)C(C)C)ccc(Cl)cc1 64901,Cc1ccc(C(=O)NCC(C)NC(C2CCCN(C(=O)OC(C)(C)C)C2)=O)cc1 64902,C1(C(=O)NC(C)Cc2nc[nH]n2)CCCCC1CNC(C1(C)CCN(C)C1)=O 64903,C1(C(=O)NCC(CC=C)(C)C)CCCN(C(C2CCC2(OC)OC)=O)CC1 64904,C(C)(c1cnn(C)c1)=CC(=O)NC(c1ccc(OCC(F)F)cc1)C(=O)OC 64905,c1(CNC(=O)NNC(=O)c2cc(I)n[nH]2)c(Br)cc(Br)c(O)c1Br 64906,CC(C(C)C(=O)N1CCOC(CNC(C2CC23CC(C)(C)C3)=O)C1)S(C)(=O)=O 64907,CC1(C(=O)NC2CC2NC(=O)CCc2nc(-c3cccs3)no2)C=CCC1 64908,c1(CC(=O)NCCC2N(C(c3c(OC)n[nH]c3)=O)CCC2)ccc(Cl)cc1F 64909,C1(C(=O)NCC(C2CC2)OC)CN(C(C2(O)CCOCC2)=O)CC(C)O1 64910,C1(C(N2CCC(OCC3CC3)C2)=O)CN(C(=O)C=Cc2ccncc2)CCO1 64911,C(=O)(CC(C)CC(C)C)N1CCN(CC(C)NC(C=Cc2ccc(C)o2)=O)CC1 64912,Cc1c(C(N2CC(Oc3cccc(O)c3)C2)=O)cc(S(C)(=O)=O)cc1Br 64913,c1(NC)cc(N2CCN(C(C)C(=O)NC(c3noc(CSC)n3)C)CC2)ncn1 64914,c1(CN(C)Cc2cn(C(C)Cc3c[nH]cc3C3CC3)nn2)nocc1C(C)(C)C 64915,n1(CC)cnc2nc(=NCC3CCCC3)[nH]c(NCC(C)CN(C)C)c12 64916,N1(C(CCSCCCC)=O)CCCC12CCN(C(=O)C(c1c(C)noc1C)C)C2 64917,Cc1nc(S)sc1CC(=O)NCC(C)(C1CC1)NC(=O)C(C1CCCCCC1)O 64918,CC(=O)CC(C)(C)CC(=O)NCCC1CCCN(C(=O)C(F)(F)CC(C)C)C1 64919,Cc1cn2c(n1)CCC(NC(=O)NCc1ccnn1Cc1ccccc1)C2 64920,c1(C(=O)NC2CC(CNC(C(C#C)(C)C)=O)C23CCC3)cccc2sccc12 64921,c1(C(=O)NC(C=CC(=O)NC(CCC)(C)CC)C)ccc2cccnn12 64922,c1(NC2CC3(CC(C)C3)C2)nccc(=NCCCCc2cnc[nH]c2=N)[nH]1 64923,C1(NC(C(C(C)C)F)=O)CCC2(CC1)CCN(C(=O)CCC1CCOCC1)CC2 64924,N1(C(CSCCC)=O)CC(NC(=O)Cc2ncoc2C)C2CCCCC12 64925,CC1CCC(CC(=O)NCCSCC(N2CCC(c3cnco3)C2)=O)C1 64926,c1(CC)conc1CC(=O)NCCOCCN(C)C(C1(OCC)CC(=O)C1)=O 64927,N1(C(c2c(C)n(-c3ccccn3)nc2)=O)CCCC(NC(=O)C2=CCSC2)CC1 64928,S(=O)(=O)(c1cccnc1N1CCC(OCCOC)C1)NCC1CCC(CC)CC1 64929,C1(NC(C2CC(NC(C=C(C)c3ccco3)=O)C2(C)C)=O)CC2CC1C(O)C2O 64930,O=CN1CCN(C(C2CC23CN(C(=O)CCc2ccc(Br)cc2F)C3)=O)CC1 64931,N1(C(C2C3(CCN(C(C4N(C)CC(F)C4)=O)C3)C2)=O)Cc2ccc(O)cc2C1 64932,CC(F)(F)C(C)(C)CS(=O)(=O)Nc1ccc2c(c1)NC(=O)CO2 64933,c1(C(=O)NC2C(CNC(c3cnn(CC)n3)=O)CCC2)cccc(OC)c1OC 64934,c1(SC)cc(C(=O)NC2(C)CC(NC(=O)CCC3(C)CCC(=O)N3)C2)oc1C 64935,c1(C(N2CCN(C(C(CC)C(C)O)=O)C(C)C2)=O)n[nH]c(C(C)C)c1[N+](=O)[O-] 64936,Cc1nc(C)n(CCC(N2CCC(C(F)F)(CNC(c3c[nH]nc3C)=O)C2)=O)n1 64937,N1(C(Cn2cnc(=N)[nH]2)=O)CCCC(CNC(=O)CCc2ccc(O)nc2)CC1 64938,CC1CN(C(=O)CC2(NC(C3CCCC(O)C3)=O)CC2)Cc2nncn21 64939,CC1OC(C)CC1C(C1CCN(C(=O)OCCCc2ccccc2)CC1)=O 64940,c1(C(=O)NC(CC)(C)CCNC(c2csc(Cl)c2)=O)cc(C)nc(O)c1 64941,Cc1ccc(C(=O)NCC2CCN(C(C3CC3C)=O)C23CCC3)c(=O)n1C 64942,C=CC(C)(O)CC(=O)NC(C)(C)CNC(=O)C(C(C)(C)O)Oc1ccccc1 64943,N1(C(c2cnc(C)s2)=O)C(CC(=O)N(CC(N)=O)CC(N)=O)C2CCCC12 64944,N1(C(C(C(C)O)(C)C)=O)CC2(CC(C(N3CCOC(C#N)C3)=O)CO2)C1 64945,C1(CNC(C(CCC)OCC)=O)CC2(CCN(C(=O)CC3CCC(C)C3)C2)CO1 64946,c1(C(C)(CO)NC(=O)NCC(c2ccccc2Cl)(C)C)cccc(Cl)c1 64947,N1(C(C2(OC)CCOC2)=O)C(C(=O)NCC2(O)CC3CCC2C3)C2CC(O)C1C2 64948,C1(C)(C(=O)NCc2cn(CC(=O)NCc3nc(C)sc3)nn2)CCC(C)C1 64949,Cc1cnc(C(=O)NC(C)C(C)(C)NC(c2cnc(=N)[nH]c2)=O)c(F)c1 64950,c1(N(C)CC2CC2(C)C)nc2ccc(S(=O)(=O)N3CCC4(C3)OCCO4)cc2s1 64951,N1(C(CN(C)CCO)=O)CCC(CNC(=O)COc2ccc(Br)cc2)C1(C)C 64952,c1(CNC2CCC(C(=O)NC(C3CCCCO3)C)C2)cc(C#N)ccn1 64953,c1(NC(=O)CSc2ccc(Br)cc2)ccc2c(n1)CCCN2 64954,c1(C(=O)NC2C(CNC(CC3C(CC)C3)=O)COC2)ccnc2[nH]ncc12 64955,N1(C(=O)NCC2CCN(c3ccccc3C(F)(F)F)C2)CCCOC(CCS)C1 64956,N1(C(C(C)S(N)(=O)=O)=O)CC2(CCC(CNC(c3ccncc3C3CC3)=O)O2)C1 64957,c1(NC(=O)CC2CCCN2Cc2cc(B(O)O)co2)c(Br)cc(F)c(F)c1F 64958,N1(C(c2ccc(C(C)=O)cn2)=O)CCC2(NC(=O)CC3CC3(C)C)CCCC12 64959,C(=O)(C(CO)C(C)(C)C)N1CCN(CCN(C(CNS(CC)(=O)=O)=O)C)CC1 64960,O=C(C#CC1CCOC1)NC1CC2CCC1CC2NC(=O)C(F)OC(F)(F)F 64961,c1(NC(c2n(C(C(=O)OC)C)nnn2)(C)CCCl)ccc2nncn2c1 64962,C(=O)(C#CC1CCCOC1)NC1CC(CNC(C2(SC)CC2)=O)OCC1 64963,c1(SC)cc(C(=O)NCCC(C)NC(=O)C(C)NC(c2cccs2)=O)ccc1F 64964,CC(CC(=O)N(C1(C(N2CCOC(C#N)C2)=O)CC1)C)C(F)F 64965,C(N=c1nc2scnc2c(N2CCC(CO)CC2)[nH]1)C1C(C)(C)S(=O)(=O)CC1 64966,c1(NC2CC(OCC)C2)nccc(=NC(CC)CC#N)[nH]1 64967,C#CC1CN(C(=O)C(C)C(CC)CC)CCN1C(=O)CCCOC(C)=O 64968,c1(C(=O)Nc2cc(OC)ncc2)nc(N=c2[nH]cnc3cc(I)sc23)cn1C 64969,c1(C(=O)NCCN(C(C2CCC(C)S2)=O)C2CC2)ccc2ccoc2c1 64970,CC(C(=O)N1CC(NC(c2ccc(CO)c(Cl)c2)=O)C2(CC2)C1)C(C)(F)F 64971,c1(C(C(=O)NC)N(C)CC2(CC)CCC2)cccc(N2CCOC2=O)c1 64972,S(=O)(=O)(c1cccnc1NC(CCO)CC(C)C)NC1(CC=C)CC=CCC1 64973,N1(C(CC2CNC(=O)O2)=O)CC2(CCC2)CC1CNC(=O)Cc1cc[nH]n1 64974,CC(C)CCCC(=O)N1CCC(O)(CCNC(C2(O)CC2)=O)CC1 64975,c1(C(=O)NCC2(O)CN(C(C3C4C5CCC(C5)C34)=O)C2)cccc2c1CCCN2 64976,C#CCCCC(C)C(=O)NC1CN(C(c2ccc(F)o2)=O)C1 64977,c1(C(N(CCCNC(=O)CC(O)C2CCCC2)CC)=O)ncccc1OC(F)F 64978,c1(N(C)C)ccnc(C(c2nnnn2C2CCC2)NC2CCN(C3CCC3)C2=O)c1 64979,CC1(C)CC(CNC(=O)CN2C(=O)CNC2=O)CN1C(C1CCC1CF)=O 64980,N1(C(C(CC)CC(F)F)=O)CC2(CCN(C(c3cccc(OC)c3)C)CC2)C1 64981,c1(OC)cc(OC)c(CNC(=O)NCC(c2ccccc2OC)(C)C)cc1Cl 64982,CC1CCCC1C(=O)NCC1(Cn2cc(-c3nccn3C)nn2)CC1 64983,c1(C(=O)NC2(CO)CCN(C(C(C)=CC3CC3)=O)C2)nccc2ccsc12 64984,C#CCC(CC(=O)N1CCC(C)=C(C)C1)NC(C1(CCC)CC(=O)C1)=O 64985,C1(CCNC(CCN(CC)CC)=O)CCCN1C(=O)CSC 64986,C=CCCC(C(=O)NCC(O)CC(C)C)NC(c1cccnc1O)=O 64987,C1(F)(C(=O)NCC(C)(C)CNC(C2(c3ccccc3F)CCC2)=O)CCCOC1 64988,c1(C(=O)NC(CC=C)CNC(=O)Cc2cncn2C)cccnc1C(F)F 64989,N=c1[nH]c2ncc(C(=O)NCC3CCN(C(=O)CCCF)C3)cc2s1 64990,c1(OCCC(=O)NCCCN(C)C(c2sc(F)cc2Cl)=O)c(F)cccc1Cl 64991,c1(C(=O)NCC2CCCC(NC(CCC#CC)=O)C2)csc2c1CCCCCC2 64992,C(C1=CCCCC1)(c1nnnn1C1CCC1)NC(c1n(C)cnc1)CO 64993,c1(C(C)(C)NCc2cn(CCC)nc2)cccc(F)c1 64994,CC1(NC(c2ccc(C3CC3)s2)=O)CCN(C(C2(C)CCOC2)=O)C1 64995,C1(NC(C(COC)N(C)C)=O)CC(F)CN(C(c2c(C3CCC3)cnn2C)=O)C1 64996,Cc1n[nH]c(C)c1CCCNC(=O)NC(c1ccc(F)cc1)C1CCOC1 64997,c1(N2CC(N(C(=O)CCc3ccc(F)cc3)C)C2)ccc(Br)cc1[N+](=O)[O-] 64998,C1(C(N(C)Cc2ncccn2)=O)CCN(C(=O)C2(O)CCOC2(C)C)O1 64999,c1(CN2CCC(CC(N3CC(OC)C(C(=O)O)C3)=O)C2)cc(Cl)c(F)c(Cl)c1 65000,CC1CCN(C(c2cc(C(F)(F)F)on2)=O)CC1N(C(=O)CCC1OCCO1)C 65001,C(C(=O)N1CCC(CCNC(C2(CO)CCC2)=O)CC1)(C(C)C)OCC 65002,c1(CC(N2CC(OC)C(NC(=O)COC(F)(F)F)C2)=O)nc2c([nH]1)CCCC2 65003,C1(C(=O)OC)C(C(=O)NCC2CCCN2C(c2csc(O)n2)=O)C1(F)F 65004,C1(C2CCCN(C(=O)C(C)C#N)C2)(NC(c2ccn(C(C)C)c(=O)c2)=O)CC1 65005,C(CN1C(=O)Cc2ccccc21)NC(c1cn(C)nn1)c1nnnn1C(C)(C)C 65006,C1(NC(C2CC(=O)N2)=O)CN(C(c2cnn(-c3ccc(F)cc3)c2)=O)CC1F 65007,Cc1oc(C)c(C(=O)N(C)CC2CCN(C(=O)Cc3nnc(O)s3)C2)c1C 65008,c1(NCC2C(NC(c3scc(C)c3Cl)=O)CCCC2)ncnc2c1cnn2C 65009,C1(CNC(c2c(CC)nc(C)[nH]2)=O)CC2(C1)CN(C(=O)Cn1nc(C)cc1C)C2 65010,C=CCN=C(NCc1cn2cccc(F)c2n1)N1CN(C)C(=O)C1C 65011,N1(C(C=CCOC)=O)CCC(C2OCCC2NC(=O)Cn2ccnc2C)CC1 65012,CCC(C(O)C(C)C)NC(=O)NCC(c1ccc(Br)cc1)(C)C 65013,C1(O)(C(C)NC(CSCCCC)=O)CCN(C(=O)Cc2ccc(C(=O)OC)cc2)C1 65014,c1(C(N(CCN(C(C(C)OC(C)(C)C)=O)C)C(C)C)=O)ccc(Br)cc1 65015,C#CCC(CC(=O)NC1CCCC(CO)C1)NC(=O)C(F)(F)CC 65016,C=CCCCC(=O)N1CC2C(NC(c3c[nH]cc3C(C)(C)C)=O)C2C1 65017,N1(C(C(CC)n2cncn2)=O)CCCCC1CCCNC(c1c[nH]c(=O)cn1)=O 65018,C1(OC)CCC12CC(C(N1CCC(C(C)NC(=O)C3=COCCC3)CC1)=O)C2 65019,CN1CC(C(=O)NCC2CCC(C(=O)NCCOc3ncccn3)CC2)CC1=O 65020,c1(COC)nn(C)cc1C(=O)N(C1CCC(=O)N1)C 65021,CCC(C)C(C(=O)NCC1=CCN(C(c2ccc(NC)cc2Cl)=O)CC1)OC 65022,C1(NC(C2(OC)CCN(C(C3CN4CCC3CC4)=O)C2)=O)CN(C)CC1(F)F 65023,c1(COC)cccc(CNC(=O)CC2CCN2C(c2ocnc2C)=O)c1 65024,c1(OC)ccc(C(C2CC2)NC(=O)C(c2ccc(C(F)(F)F)cc2)O)cc1C 65025,N1(C(C2(CSC)CC2)=O)CCOC(C2CN(C(C3CN(C(C)C)C3)=O)C2)C1 65026,c1(C(N2CCN(C(c3c(C)ncc(C)c3)=O)CC2C)=O)cc(C)ccc1[N+](=O)[O-] 65027,c1(C(=O)NCC(=C)CCNC(c2c(C)nn(C)c2C)=O)sccc1S(=O)(=O)NC 65028,N1(C(C=CCCC)=O)CCCC(C)(CNC(=O)CCOc2ccccc2Br)C1 65029,n1(CC(=O)NCC(COC)NC(=O)Cc2cn(C)nc2C)cccc(C)c1=O 65030,C=CCC(CC)C(=O)NCCC1CC(NC(=O)Cc2cccc(NC(N)=O)c2)C1 65031,C(=O)(CCC(C)NC(C1(C#N)CC=CC1)=O)NCC(CSC)OC 65032,C1(c2ccc(F)cc2)(C(=O)NCC2(OC)CN(C(C(CC)C)=O)C2)CCOCC1 65033,CCC1c2cc(Cl)cc(Cl)c2CCN1Cc1cnc(-c2ccccc2)o1 65034,C(CNC(=O)CCc1nc[nH]n1)(C(=O)N(C)C(C1(C)CC1)C)OC 65035,CC1(CCNC(=O)C=CC2CC2)CCN(C(=O)CNC(=O)Oc2ccsc2)C1 65036,C(C(C(=O)N(C1CC1C1CC1)C)NC(=O)Cn1cc(C)cn1)OCC 65037,c1(N2CCN(C)C(CO)C2)nc(N2CCCC(c3nncs3)C2)nc2c1CCC2 65038,C1(CC)(CO)CCN(C(C2(C)CCCN2C(c2nccnc2N)=O)=O)CC1 65039,CC1Cc2ccccc2N1CCNC(=O)NC1(C(=O)O)CC(C2CCC2)C1 65040,CC(C)C(O)CC(=O)N1CCN(C)C(C(=O)NCC2CCCCS2)C1 65041,c1(CNC(CN(C(C)=O)C)=O)cnn(C)c1C(=O)NCCC1CCCC(C)C1 65042,N1(C(c2c(C)nc(O)cc2)=O)CCCCCCC1C(=O)NC1C2CCCC12 65043,C1(NC(c2cc(C(C)C)no2)=O)CCCCCN(C(=O)C(=Cc2c[nH]cn2)F)C1 65044,c1(OC(C)C(=O)NC2CN(C(C3C4COCC34)=O)CCC2O)ccc(C#N)cc1 65045,c1(CN2CCC(F)(C(=O)Nc3cc(C)c(I)cn3)C2)cccc2cccc(C)c12 65046,C1(NC(COCC#C)=O)CC2(C1)CN(C(c1csc(C3CC3)n1)=O)C2 65047,S(=O)(=O)(c1c(F)cccc1F)NC1C(C(=O)Nc2cncc([N+](=O)[O-])c2)C1 65048,CS(=O)(=O)c1ccc(S(=O)(=O)NCCNC(=O)Nc2ccc(Cl)c(Cl)c2)cc1 65049,c1(C(=O)NCC2CCCCC2)ccc(NC2=NCCC2)cc1 65050,c1(C(C)C)cnc(C(c2nnnn2C2(C)CC2)NCc2nc(C(N)=O)cs2)[nH]1 65051,C=CCC(CC(=O)Nc1cnc(C2CC2)nc1)NC(C1CC(CC)=NO1)=O 65052,c1(C(=O)NC(C(CO)NC(C(CCCOC)C)=O)C)nnc(O)c2ccccc12 65053,C(=O)(CC(C)P(C)(C)=O)N1CCC(CCNC(c2cc(C)nc(O)c2)=O)C1 65054,Cn1c(C(=O)NCC2(C(F)F)CCN(C(c3cn(C4CC4)cn3)=O)C2)cnc1O 65055,C1(CN(C)C)CC(O)CN1C(c1n[nH]cc1CNC(=O)CC1CC(=O)C1)=O 65056,n1(CCC)ncc(C(N2CCCCC2CCNC(C2CCS(=O)CC2)=O)=O)c1Cl 65057,C1(CNC(CC(C=C)CC)=O)CC2(CCN(C(=O)C(C)C(C)CC)CC2)CO1 65058,COn1cnc(C)c1C(=O)NCC1CCC1NC(c1cc(F)ccc1C1CC1)=O 65059,c1(C(N(CCN(C(C(C)OCC)=O)C)C(C)C)=O)cc(S(C)(=O)=O)oc1C 65060,C#CCCCCC(=O)N1CCC(NC(=O)CCc2cccc(OC)n2)C(F)C1 65061,N1(C(c2c(CC)nco2)=O)CC(NC(C2CCCC2C(C)C)=O)C(C)C1 65062,c1(C(N(C2CCN(C(CCCC)=O)C2)CCO)=O)c(C)cccc1C 65063,c1(C(=O)NC(C2CCCN(C(C3(COC(C)C)CC3)=O)C2)C)cc(Cl)ncc1O 65064,c1(C(=O)NCCCNC(c2cc(C(=O)O)ccc2O)=O)cc(Cl)c2n[nH]cc2c1 65065,CCC(C)CC(=O)N(C1CC(NC(=O)Cc2sc(C)nc2C)C1)C 65066,C(=O)(CC1CCc2ccc(O)cc21)NCC(C)NC(c1cccc2cncn12)=O 65067,n1(CC)nc(C)cc1C(=O)NCC1CN(C(=O)C(C(C)C)NC=O)CC1O 65068,N1(C(Cc2c(C)cnn2C)=O)CCC2CC2(C(=O)NCC2(O)CC=CC2)CC1 65069,Cc1[nH][nH]c(=N)c1C(N1CCC(CNC(c2cnc(Cl)[nH]2)=O)C1)=O 65070,N1(C(C2(C#C)CN(C(C3CCC(F)(F)C3)=O)C2)=O)CCN(C)CC1C 65071,C1(C(=O)NCC2(F)CCCN(C(=O)C(C)C(C)C)C2)(CC)CCC(O)CC1 65072,C1(CN(C(=O)CC(O)c2ccccc2)CC)CCCCN1C(c1cnc[nH]1)=O 65073,c1(C(=O)NC2CCN(C(c3ccc(N)cc3Br)=O)C2)occ2c1CCOC2 65074,CCC(C(=O)NC(CC1CCC1)C(=O)NCCCCCSC)N(CC)CC 65075,c1(OC)cc(NCC=CCNC(=O)Cc2nncn2C)c(Cl)cc1[N+](=O)[O-] 65076,C1CC(=O)NOC(C)C(=O)N1CC#C.C(CC(=O)OC)OCC#C 65077,Cc1cc(C(=O)NCC(C)NC(=O)C(O)C2CC2)c(C)n1CC(F)(F)F 65078,n1(CC)nc(C(=O)NC2CN(C(=O)CSC3CC3)CC2C)cc1C1CC1 65079,c1(CC(=O)N(CCNC(C(C)OCC(C)C)=O)CCOC)ccc(CC(C)C)cc1 65080,C(=O)(C#CC(C)(C)CNC(C1(C)CCCC1O)=O)NC(C(=O)N(C)CC)C 65081,C(=O)(C(C)C(F)(F)C(F)F)N1CCN(C(CC2CCC(C)CO2)=O)CC1CO 65082,C1(C(=O)NCC2CC(NC(C3CCS3(=O)=O)=O)C2)CCC([N+](=O)[O-])CC1 65083,c1(NC(C2CCC(C)(C(C)(C)C)C2(C)C)=O)cccc2c1COC(=O)N2 65084,c1(C(N2C(CC(C)C)CCCC2)C(=O)NC2COC2)cccn2ccnc12 65085,N1(C(C(CC)F)=O)CC2(C)CC1(C(=O)NC(C)C)C2 65086,N1(C(C(CCC)C)=O)CCN(C(=O)CSCC(C)C)CC1C 65087,N1(C(C(COC)OC)=O)CCN(C2CN(C(C3COCCN3C)=O)C2)CC1 65088,C1(C(C)(C)O)(CNC(=O)CC2CCC2)CN(C(=O)C=CC2CCCC2)C1 65089,N1(C(c2cc(CC)on2)=O)CCN(C(=O)C=Cc2ccc(SC)cc2)C(CF)C1 65090,c1(N(C)C)ccc(C(=O)NC2CC(C(F)F)(NC(=O)COC3CC=CC3)C2)cc1 65091,c1(C(C)NC(N2C(C(=O)NCCN(CC)CC)CCC2)=O)ncccc1F 65092,N1(C(C(CC)C)=O)CCN(C(=O)C=Cc2ccc(OCC#N)cc2)C2CCC12 65093,Cc1cc(C(c2nnnn2-c2ccc(F)cc2)NC2(CCF)CC2)c(C)cc1Br 65094,Cn1cnc2ccc(C(N3CCN(C(c4ccon4)=O)C(C(F)(F)F)C3)=O)cc12 65095,CC1(NC(C2C3CC4C(C3NC(c3cnc(O)o3)=O)C24)=O)CCCCCC1 65096,C1(C)(C(=O)NCC2(OCC)CCC2)CC(OC)CN1C(=O)CCC(C)C 65097,Cc1cc(C(=O)NC2CCC2NC(=O)CCCCCN(C)C)c(C)n1CC1CC1 65098,C1(C(C)NC(=O)CC2(O)CCCOC2)CCN(c2nnc(C(F)F)s2)CC1 65099,C1COC(C)(C)C1.CCC(C(=O)NC(CC(N)=O)c1cn(CC2CC2)nn1)N(C)C 65100,c1(C(=O)NCCC2CCC(NC(=O)Cc3cccs3)C2)cc(F)c2c(c1)CCC2 65101,c1(C(=O)NCC(C(=O)NCC(COC)O)N(C)C)ccc(C)nc1O 65102,C1(C(N(CC(C)NC(C2(CC)CCC2)=O)C)=O)CCCN(c2ccnc(Cl)n2)C1 65103,C(C(F)(F)C(=O)NCCN(C(c1cc(-c2cccnc2)on1)=O)C1CC1)OC 65104,C(CN=c1[nH]c2ccc(F)cc2o1)NC(C1CCN(C(C(C(C)O)C)=O)CC1)=O 65105,C1(NC(C2C3CN(C(C(C)=C4CCCC4)=O)CC32)=O)CCCOC12CCC2 65106,c1(C(N2C(C)CCC(CNC(=O)Cc3cccs3)C2)=O)cncc2c1CCC2 65107,N1(C(C(C)=CC2CC2)=O)CCCC(CO)(NC(c2cncc(Cl)c2)=O)C1 65108,C#CC1CN(C(C2C3CN(C(c4cnc(Cl)n4C)=O)CC23)=O)CCO1 65109,c1(C(=O)NC2(CF)CCN(C(C(C=C)O)=O)C2)cccc2c1COC2 65110,C1(NC(C2CN(c3ccc(C)cc3)C(=O)C2)=O)CC2(CCC(C(=O)O)CC2)C1 65111,C(CCC(C)(C)C(=O)N1CC(O)C(O)CO1)NC(c1c(OC)scc1)=O 65112,Cn1[nH]nnc1=NCC1(c2ccccc2)CCCN1C(=O)C(=O)NC1CC1 65113,N1(C(c2cnc3sccn23)C(=O)NCCCC)CCC2(COC(C)C2)C1 65114,N1(C(CCC2C(=O)NC(=O)N2)=O)CC2CCN(C(C3CC=CC3)=O)CCC2C1 65115,c1(CN2CCN(CCOC)CC2)ccc(-c2ccc(Cl)s2)cc1F 65116,c1(OC)cc(C(N2CC(O)CC2CNC(=O)COC(C)=O)=O)c2c(c1)CCO2 65117,C1(NC(CNCC(=C)C)=O)CCOC12CCN(C(=O)CCNC(=O)COC)CC2 65118,N1(C(C(F)=CCC)=O)CC2CC1CN(C(c1cc(C)ccc1Cl)=O)C2 65119,CCC(C(=O)NC(C1CCN(C(C2CCN(CC)C2)=O)C1)(C)C)n1cncn1 65120,c1(C(N(CC(=O)NC)CC)=O)ccc(C2COCCN2Cc2ccsc2Cl)n1C 65121,C1(C(N2CC(CC=C)(NC(=O)C(C)OCCCC)C2)=O)CCOC(C)C1 65122,CN1CCOC(C(=O)NC2CN(C(c3cc(-c4ccccc4)ns3)=O)CC2O)C1 65123,N1(C(CC(=C)Br)=O)CCN(C(=O)Cc2cccc(OC)c2Cl)CC(O)C1 65124,C1(CN(C2CCN(CCS(N)(=O)=O)CC2)C)CN(C(=O)OC(C)(C)C)CC1O 65125,c1(CC)occc1C(=O)NC(CNC(c1cnc(C)s1)=O)CCOC 65126,C1(CCN(C(C)C)C(C2(NC(=O)COCC3CCCC3)CC2)=O)CCC2CC2C1 65127,N1(C(C)C)CCC(C(=O)NC(C)CC2CCN(C(=O)CC=C(Cl)Cl)CC2)CC1 65128,C(=O)(CC(O)Cc1ccccc1)N1CC(NC(C2CSC2)=O)C1 65129,n1(CCNC(NCC2C(CC)C2)=NCCC(C)=O)nnc2ccccc2c1=O 65130,c1(C(=O)NCCN(C(=O)C(C(C)CC)OC)CCC)cc2cc(Cl)ccc2n1C 65131,c1(NC(C2CCCN(C(C3COC(C)(C)C3)=O)C2)C)ncc(I)cn1 65132,c1(CC)cccc(C(N2CC(C)C2C(=O)NCc2ncsc2C)=O)c1 65133,c1(C(=O)NC2CCN(C(C3(OC)CCOC3)=O)C2)cc2cccc(Cl)c2nc1C 65134,c1(OC(C)C(N2CCCCC2CCCNC(=O)CP(C)(C)=O)=O)cccc(F)c1 65135,C1(CNC(C(C)(C)c2ccccn2)=O)CN(C(C2CCCS2)=O)CCC1(F)F 65136,c1(-c2nc(C3C(C)(C)CN3)on2)cc(Cl)cn2nccc12 65137,c1(C(=O)OCC)cc(C)sc1NCc1cn(-c2ccccc2OC)cn1 65138,C1(CNC(c2c(C)cn(C)c2)=O)CN(C(c2ocnc2C2CC2)=O)CC(C)(C)C1 65139,C(CCCCCC(=O)N1CC2CC=CC1C2)NC(c1nccc(Cl)c1F)=O 65140,C1(C(N(CCCN(C(=O)CCn2cnnn2)C)C)=O)CCCNC1=O 65141,C1(C(=O)Nc2ccsc2)C2CN(C(=O)CCCOC3CCOCC3)CC12 65142,c1(C(=O)NCC2CN(C(C(CC(C)C)OC)=O)CC2(F)F)scc2c1OCCO2 65143,c1(C(N2CC(C)N(C(=O)C=CC3CCOC3)CC2)=O)cc(Cl)c(F)c(Cl)c1 65144,CC1N(N2CCOC(c3noc(-c4ccccc4)n3)C2)C2CCCOC12 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65321,c1(NC(C2N(C(C(C=C)OC)=O)CCC=C2)=O)cc(C)ccc1CO 65322,C1(C(=O)NCC(CSC)OC)CCC(C)(C)N(C(=O)C2=C(C)OCCS2)C1 65323,N1(C(CC(=C)C)=O)CCCC2(CCCN2C(c2cnn(C)c2OC(C)=O)=O)C1 65324,CC(C)CC(C)C(=O)NC1C2CCN(C(c3ncnc(O)c3Br)=O)C12 65325,c1(CC(=O)NC2CN(C(C(CSC)O)=O)C(CO)C2)c(C)cccc1C 65326,C1(NC(c2c(C)cnn2C)=O)CCOC2(CCN(C(c3ccoc3Cl)=O)CC2)C1 65327,C1(C2CCN(C(=O)CC(=O)OC)CC2)(NC(C2CC(N(C)CC)C2)=O)CC1 65328,S(=O)(=O)(c1c(F)cccc1F)N(c1ncnc2[nH]ccc12)c1ccc(=N)[nH]c1 65329,C1(C)(COC)CN(C(c2cc(CNC(c3cnc(Cl)s3)=O)[nH]n2)=O)C1 65330,C#CC(C)(C)C(=O)N1CC(C=C)(CC(=O)NCCc2ccc(F)cc2)C1 65331,c1(C(N2C(C)CC(NC(=O)CCc3nnc(O)nc3O)C2)=O)ccc2ccnn2c1 65332,CCCC(C)(C)CC(=O)NCC1(OC)CN(C(c2nc[nH]c2C(F)(F)F)=O)C1 65333,C=CCCC(C(=O)N1CCOC(CO)C1)NC(c1cccc(OC)n1)=O 65334,c1(C(N(C)CC2N(C(C(C)N3CCC3)=O)CCC2)=O)ccnc(C(F)(F)F)c1N 65335,c1(C(C)(F)F)ccc(CNc2csc(-c3cccc(Br)c3)n2)nc1 65336,c1(C(=O)NC(C)CNC(=O)CSC2CCOC2=O)cncc2c(O)nccc12 65337,C1(C(=O)NCC(CNC(C2(C=C)CCCC2)=O)(C)O)CCC2(CC1)OCCO2 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65355,C(=O)(C(F)(F)CCn1cccn1)NCC12C(CN(C(CC3C(C)OCC3)=O)C1)C2 65356,C12(CNC(c3ccnnc3O)=O)CCCC(CN1C(C1Cc3nncn3C1)=O)C2 65357,c1(C(N2C(CNC(C34OCC(COC)(C3)C4)=O)CC2)=O)csc([N+](=O)[O-])c1 65358,C(=O)(C(CC(C)C)C(C)C)NC12CN(C(c3cc(C)ncc3C)=O)C(CC1)C2 65359,Cc1c(C(=O)NC2CN(C(C3CC3F)=O)CCC2O)oc(=O)c2ccccc12 65360,c1(N(C)C)cccc(NC(C2CN(C(=O)CSCc3cccs3)CCO2)=O)c1 65361,C1(CC(=O)N(CCCCCC)CCNC(=O)CCCOC)CC(OC)C1(C)C 65362,c1(C(N2CCC(NC(CCC(CC)OC)=O)C(O)C2)=O)nn(C)c2c1COCC2 65363,C1(NC(c2ccon2)=O)CCCCC1OCc1cn(C2CCSCC2)nn1 65364,c1(N2CCC(c3cccc(C)c3)C2)nc2ccccc2nc1NCCC(C)C(F)F 65365,C(=O)(C1=CCC(C)(C)CC1)NCCC(C(=O)NC1CCOCC1C)OC 65366,C12(C(N(C(C)CNC(C3COC(C)(C)C3)=O)C)=O)CCC(C(F)(F)F)(CC1)CC2 65367,C=CC(C)(CC)C(=O)NCc1cc(C)c(C(=O)N(CC(O)CO)C(C)C)o1 65368,CCC(CNC(=O)CC1CCCC1O)(CC)C(=O)N1CC(N2CC(O)C2)C1 65369,CCC(CC(=O)NC1(CO)CCCN(C(C)=O)C1)CC(F)(F)F 65370,N1(C(c2c(CC)occ2)=O)CC2CC2(CNC(=O)CCCN2CCCC2)C1 65371,c1(NC(C2(CNc3cc(CC)ncn3)CC2)=O)ccc(Br)c2ncccc12 65372,N(C(=NCCC(C)=O)NCC1CCCC1CCC)Cc1n(CC)ncn1 65373,C(=O)(C1=C(C#N)CCC1)N1C(CNC(CC(C=C)CC)=O)CCC1 65374,C(C(C)(C)CCNC(=O)CC1COCCO1)NC(C(C1CC1)OCC)=O 65375,C1(C(=O)OC)CCCC(NC2CCCC(c3ccccc3)C2)CC1 65376,c1(C(N2CC(CNC(c3oc(C)c(CO)c3)=O)C2)=O)cc(O)ccc1Br 65377,CCCCCCCCCC(O)C(=O)N(CC(C)CNC(c1nccnc1C)=O)C 65378,C12(C(=O)NCc3nc(C)c(C(=O)NCC4CC(F)C4)o3)CCCC1C2(F)F 65379,C1(NC(c2cn(CCC)nc2)=O)CCN(C(=O)CCCCC(N)=O)CCC1(F)F 65380,CC(C)CC(C)CNC(=O)C(O)CNC(=O)CSC(F)(F)F 65381,N1(C(CCCC#C)=O)CC(CCNC(c2cnc(OCC)c(Cl)c2)=O)OC(C)C1 65382,N1(C(c2c(C)[nH]c(=N)s2)=O)CCC2(C1)CN(C(=O)C(C)(C)C(F)(F)F)CC(C)O2 65383,c1(CC)cccc(CC)c1C(N1CC(F)CC1C(=O)NCCCS(C)(=O)=O)=O 65384,C1(NC(CCC=CCC=C)=O)CC(C)N(C(=O)CSc2cn[nH]c2)C1 65385,CS(=O)c1ccccc1C(N1CC2(C1)CN(C(c1cnc(F)c(Cl)c1)=O)C2)=O 65386,C1(C(=O)NCCC2CCCN(c3ccnc(C)n3)C2)CCCC(C)(C)C1 65387,Cn1cnc(CCC(=O)NCC(CNC(c2cc(C3(C)CC3)n[nH]2)=O)CO)c1 65388,c1(C(=O)NC(C)CN(C)C(C2CCCN2c2cnccn2)=O)ccc(Cl)cc1O 65389,CCCS(=O)(=O)C(C)C(=O)NC1CCCC1NC(c1cnc2n1CCCC2)=O 65390,C1(C(=O)NC(CNC(=O)Cc2sccc2Cl)C2CC2)CC=CC(O)C1 65391,C1(C(=O)Nc2cccc(CCCC(=O)OC)c2)CCC2(CCCC2)C1 65392,C(C1=CCN(C(=O)C(C)S(C)(=O)=O)CC1)NC(CCCc1scc(C)n1)=O 65393,N1(C(Cc2n(C)ncc2)=O)CC(=O)NCC1C(=O)NCCOCCN=[N+]=[N-] 65394,C1(N(CCOC)C)CCOCC1NC(C1(N(C(=O)CCC2CC2C)C)CC1)=O 65395,C1(NC(c2ccc(CN(C)C)o2)=O)C2CC1CN(C(c1nnsc1C(F)F)=O)C2 65396,C1(CC)C(C)CCN1C(=O)CN(C(c1ccnn1COC)=O)CCF 65397,C1(CNC(C2CC(OC)C2)=O)N(C(c2ccc(Cl)cc2Cl)=O)CCCC1(C)C 65398,c1(NCCN2C(C)CCC2)cc(NCCN2CCOCC2)ncn1 65399,C1(NC(C(C)NC(COC)=O)=O)CN(C(C2CC(C)(C)C2)=O)CCC1C(F)(F)F 65400,CC(O)C(C(=O)NCC(C)(C)OCCNC(C12CC(C)C1C2)=O)NC(N)=O 65401,C#CCC(C)(CC)C(=O)NCC(C(=O)N(C)Cc1nc(C)ns1)C(C)C 65402,N1(C(C(C)N=[N+]=[N-])=O)CC(C)C(C)(C(N2CC(C)(N(C)C)C2)=O)C1 65403,CCC(F)(F)C(=O)NCC(C)(C)CNC(=O)CN1CCNC(=O)C1 65404,C(C)(C(=O)N1CCC1CNC(=O)C(C)=CC1CC1)NC(=O)NC 65405,C1(C(=O)OC(C)(C)C)CCCC2(CN(c3ccc([N+](=O)[O-])c(Br)c3)C2)O1 65406,c1(C(N2CC(NC(C3CCC3n3cccn3)=O)C(CO)C2)=O)ccc(F)cc1F 65407,C1(NC(C2C(C=C)OCC2)=O)CCN(C(=O)CC(C)C2CCCCC2)CC1O 65408,C1(C(=O)OC)CN(C(=O)Cc2cnc(Cl)cc2C)CCC1CN 65409,CC(C)(CC(=O)N1CC=CC(NC(C2CCCC3CC23)=O)C1)c1ccccc1 65410,c1(C(=O)NCC2CCN(C(C(C(C)C)OCC)=O)C2)cccc2nc[nH]c12 65411,C(Cn1cc(CCCN(C)C)nn1)(CC(C)C)OC.c1(C2C(=O)N2)ccccc1 65412,c1(NC(c2cnn(C)c2Br)c2n(C(CC)C)nnn2)cc(Br)c(O)nc1C 65413,N1(C(c2cc(CNC(CCC(C)C)=O)[nH]n2)=O)CCC(O)C12CCC2 65414,c1(CC(C(C)C)NC(=O)NCC2CC(F)CN2)ccccc1C(F)(F)F 65415,C(=O)(C1=COCCO1)NCCOC1(CNC(C(CC)F)=O)CCOCC1 65416,C1(Nc2nccc(N3CC(CCC)OCC3)n2)Cc2ccccc2C1OC 65417,c1(OCC(C)C)cc(C(=O)NC2CCC2CNC(=O)C(C2CC2)N(C)C)ccn1 65418,C1(C)(CNC(C(C)N2CCC2)=O)CC(F)(F)CN1C(=O)C=Cc1ccc(F)nc1 65419,C1(O)(CN(C(Cc2cc(C)sc2)=O)C)CCN(C(=O)CC(C)N(C)C)CC1 65420,Cc1cc(NC(=O)CN(C)C2CC2)ccc1NC(=O)CCN1CCCC(C)C1 65421,C(=O)(CC(O)CNC(C1CS(=O)C1)=O)NC(c1scc(C)n1)C 65422,c1(C(N(CC2=NOCC2)C)=O)ccccc1OCc1ccc(F)cc1 65423,C=C(Cl)CC(C(=O)NCC(=C)C)NC(C1C=CCS1)=O 65424,C=CC(C)CC(=O)NCC1CC1CNC(=O)C(c1ccn(C)c1)C 65425,N1(C(C(c2ccccc2)SCC)=O)CC2C(CNC(C3CCOC(C)C3)=O)C2C1 65426,c1(C(=O)NCC(C)NC(=O)C(C)Cc2ccncc2)cnc2ccccc2c1 65427,C1(CNC(c2nc(C)oc2)c2nnnn2CCCF)CN(C)CCO1 65428,C#CC1(C(=O)NCCCc2ccccn2)CCN(C(c2ccc(Cl)cn2)=O)C1 65429,C=CCC(F)(F)C(=O)NCC(C)(C)CC1CN(C(C2C(F)(F)C23CC3)=O)C1 65430,CC(CC(=O)N1CCCCC1c1n[nH]cc1NC(c1ccccc1)=O)C(C)(C)C 65431,C1(C(CC)C)CCCCN1C(c1cc(CO)ccn1)C(=O)NCc1cccs1 65432,C1(CC=C)(NC(=O)CN2CC(C)(OC)C2)CCN(C(=O)Cc2csnc2C)C1 65433,N1(C(c2c(Cl)nn(C)c2Cl)=O)CCC2CN(C(=O)C3=COCCC3)CCC2C1 65434,C(=O)(C(CC)(CC)CO)N1CC(CC)C(NC(c2snnc2C)=O)C1 65435,CN1CCN(C(C2CN(C(=O)C(C)(C)O)CC(C)(C)C2)=O)CCC1=O 65436,C1(C(N(CCCNC(C(C)OC(C)(C)C)=O)C)=O)CCC(O)C1 65437,N(C1CCSc2ccc(Cl)cc21)C(c1nnnn1C1CC1)CCn1c(C)nnc1 65438,C(CCCCC(=O)NC1CCN(C(=O)COCCCC)C(C2CC2)C1)=CC 65439,c1(C(N2C(CC(=O)NC3CCN(CC)C3)CC(O)C2)=O)ccc2[nH]nc(Cl)c2c1 65440,c1(CSCCNC(Cn2c(CC)ncc2)=O)cccc(N)c1C 65441,C1(NC(CSCc2ccc(C)cc2)=O)CC(NC(C2(C3CC3)CC2)=O)C12CCC2 65442,c1(CC)ccccc1C(N1CC2CC2(NC(=O)C(C#N)C2CC2)C1)=O 65443,c1(C(N2C(CNC(CC(=O)NC)=O)CC(F)(F)C2)=O)c(C)nc2ncnn2c1C 65444,c1(OC)ccc(C(N2CCC3CCC23)C(=O)NCC2CC2)c(Cl)c1O 65445,C(C(C)(C)C(=O)N(CC(O)CN(C(=O)CN1CCS(=O)CC1)C)C)OC 65446,N1(C(CC2C(C)=NNC2=O)=O)CC2(C=C(C(=O)NCc3cccnc3F)CO2)C1 65447,c1(C(=O)NC(C(=O)NCC2CC3(CC3)C2)C2(C)CC2)cnc(C2CC2)nc1 65448,c1(C(=O)NC(C2(O)CCN(C(=O)C3=C(Cl)CC3)CC2)C)ccc(Cl)c(Cl)c1 65449,c1(CC)cccc(C(N2CCC(O)(CCNC(c3ccc(CO)o3)=O)C2)=O)c1F 65450,C(=O)(C(C#N)C(C)(C)C)N1CC(C(N2CC(SCC)C2)=O)C(F)C1 65451,N1(C(c2c(CC)ocn2)=O)CCCC(N(C(=O)CC2(O)CCCCC2)CCO)C1 65452,Cc1cc(CN2CCC2(C)C(=O)Nc2cc(F)c(F)cc2I)c(O)c(C)c1 65453,CC(C)(C)S(=O)(=O)CC(=O)N(C1CCCCC1)CCNC(=O)C(F)C(F)(F)F 65454,C1(NC(C2CC3C=CC2N(C(c2cnc(Cl)s2)=O)C3)=O)CN2CCC1(F)CC2 65455,C(=O)(C(C(C)NC(c1ccc2[nH]ccc2c1)=O)C(C)C)NCC(CC1CC1)OC 65456,Cc1cnc(C(=O)NC2CC3CC2N(C(c2nc(Cl)ccc2N)=O)C3)cc1C 65457,N1(C(C2(C#N)C(C)(C)C2)=O)Cc2[nH]nc(C(=O)NC3CCN(C(N)=O)C3)c2C1 65458,CC(C)(C)C(CNC(=O)C(C)(C)c1ccc(Cl)s1)NC(c1cn(C2CC2)nn1)=O 65459,c1(COC)nc(Cl)cc(=NCC2(CNC(c3c(OC)ncnc3C)=O)CCC2)[nH]1 65460,CCCCC(C(=O)NC(C(N1CC2(CCC(=O)NC2)C1)=O)C(C)OC)C(C)C 65461,CCC(CC(=O)NOCC(=O)NCC1CCC(=O)O1)CC(C)C 65462,c1(OC)cc(Br)ccc1C(c1nnnn1C(C)C)NCc1cccc(Br)c1 65463,c1(NC(C(N2CCC(C)(C)C2)=O)=O)ccc(F)c(S(=O)(=O)N(C)C)c1 65464,CCC1=NOC(CNC(C2CCC(NC(=O)Nc3cn(C(C)C)nn3)CC2)=O)C1 65465,N1(C(COC(C)C)=O)CC2CCN(C(=O)CCCF)CC12 65466,C#CC(CNC(=O)CC1CCN1C(=O)CCc1cscn1)CC 65467,c1(C2(C(=O)NC3CN(C(c4c(C)[nH]cc4)=O)CC3F)CC2)ccc(Cl)c(F)c1 65468,N1(C(c2cc(CC)[nH]n2)=O)CCC(C2CC2)C1CNC(=O)CSCC#N 65469,c1(C(N(CC(CC)NC(c2occc2C)=O)C)=O)sccc1Cl 65470,c1(NCCC(CCC)O)ncc(C)cc1S(=O)(=O)NCC#CCCO 65471,c1(C(=O)OCC)cccc(-c2nc(N(C)Cc3nnnn3C)n(C)n2)c1 65472,c1(CC(=O)NCC(CC(C)C)NC(=O)C2CC2)ccc(S(=O)(=O)N2CCCC2)s1 65473,Cc1oc2cc(C(N3CCC(C)N(C(=O)CC4(C)CC4(F)F)CC3)=O)[nH]c2c1C 65474,N1(C(C2N(CC)CCC2)=O)C2CCC(C(=O)Nc3ccc4occc4c3)C1CC2 65475,N1(C(C(C)SC)=O)CCN(C(c2cc3n(n2)CCN(C)C3)=O)CC(C)(F)C1 65476,c1(-n2cc(C3(O)CN(C(C4N(C(C)C)CCCC4)=O)C3)nn2)cccc2ccnn12 65477,C1(CN(C(c2nnc(-c3ccccc3)s2)C(=O)NCC(F)F)C)CCCSC1 65478,c1(C(N2CCC(NC(C3(C)CC=CC3)=O)C2)=O)cc(F)c(Br)c(Cl)c1 65479,CC(C(C)C(=O)NCC(F)F)NC(C1COC(=O)N1C)=O 65480,c1(C(=O)NCC(C(=O)NC(C)(C)CCO)CC2CC2)n[nH]cc1[N+](=O)[O-] 65481,C1(C(=O)NC23C(CN(C(Cc4ccn(CC)n4)=O)C2)C3)CN2CCN1CC2C 65482,C12(C(=O)NCC(CC)NC(c3cc4sccc4cn3)=O)C3CC(CC13)C2(F)F 65483,c1(CC(C)C)ccnc(NC(=O)CSc2ncccc2F)c1 65484,N1(C(C2CN(C(C3=NOC(C)C3)=O)C(C)(C)CC2)=O)CC(C)C12CCOCC2 65485,Cc1cc(C(=O)NC2CN(C(=O)C#CC3CCCOC3)C2)cc(S(C)(=O)=O)c1F 65486,C(c1ccccc1OC)=CC(=O)NCC(=C)CCNC(c1cnsn1)=O 65487,c1(CC(N2CCC(O)(CNC(CCS(C)=O)=O)C2)=O)ccc2c(c1)OCO2 65488,CCN=c1ccc(C(N2CC3CC2C3CNC(C2OCCN(C)C2=O)=O)=O)c[nH]1 65489,CC1CN2CCN1CC2C(=O)NCC1CCCCN1C(c1cnco1)=O 65490,C(C)(C(C(=O)N(C1CN(C(C)C)C1)C)C(C)C)NC(Cn1nnc(C)n1)=O 65491,c1(CC)ccsc1C(C(=O)NCc1ccco1)N(CCF)C1CC1 65492,C(=O)(C(C(C)C)C(C)C)NCC1(OCC)CN(C(C2OCCC2C)=O)C1 65493,c1(C(=O)NC2CCN(C(C3CC(SC)C3)=O)C2)cn(C)nc1C(C)(C)C 65494,c1(C(C(N2CCCC(NC(C(CCC)NC(C)=O)=O)C2)=O)O)cc(Cl)cc(Cl)c1 65495,C(N=c1[nH]c2c(c(=NCCCN3CCC(F)(F)CC3)[nH]1)SCC2)C1(C)CC1 65496,Cc1cnc(C(N2CCC3(CC3C(=O)NCCOCC(F)F)C2)=O)c(C)c1 65497,N1(C(CCSCCC)=O)CC(CNC(=O)C(C)Cc2ccco2)(COC)C1 65498,c1(NCC(C)N(C)C(c2cc(F)c(CO)c(F)c2)=O)ncccc1S(C)(=O)=O 65499,C(C)(C(CC(=O)NCCOC1CC1)NC(C1CC(C(C)C)=NO1)=O)OC 65500,C1(CC(=O)NC(C(=O)N(CCCOC)C)Cc2cn[nH]c2)CC(=O)NC1=O 65501,n1(CCC(=O)NCCC(C)NC(CC(=C)C)=O)c(=O)n(CC)c2ccccc12 65502,c1(OC)c(C(=O)NC(C)(CNC(=O)CC2(NC(C)=O)CC2)CO)csc1Cl 65503,CC1C(NC(C2CCCCC2O)=O)CCCN1C(C1CC(=O)N1)=O 65504,CNS(=O)(=O)N1CCN(Cc2ccc(OCC(F)(F)F)nc2)CC1 65505,N1(C(C(CNC(c2cnn(CC)n2)=O)(C)C)=O)Cc2ccc(C)cc2C1 65506,c1(CC)cccc2c(C(=O)NCC(C)NC(=O)C(C)(C)C3CCOCC3)c[nH]c12 65507,c1(CC)c(C(=O)NC(C)CNC(=O)CO)nnn1CC 65508,CC(C)C(CN1CCCS1(=O)=O)C(=O)NCCCN(C)C(c1scnc1Cl)=O 65509,C1(NC(CCN2CCN(C)CC2)=O)COCCN(C(C2CCCCN2C)=O)C1 65510,N1(C(CC2(C#N)CCC2)=O)CCCC(NC(=O)COCCCF)C1 65511,CN1CC=C(CC(=O)N2C3CCCC2CC(NC(=O)CC2(C)CCCO2)C3)CC1 65512,CCC(C)(C)C(O)C(=O)NCCC1(C(=O)NC2CC3(CCCO3)C2)CCCC1 65513,C1(C(C)C)(C(=O)NCCN2CCC(CO)C2)CCCN1C(=O)CN1CC(C)(C)C1 65514,c1(C(=O)NCC2CCN2C(c2cccc(F)n2)=O)ccc2cc[nH]c2c1 65515,C1(C(=O)NC(CNC(c2cc(COC)on2)=O)C2CC2)(CO)CCCNS1(=O)=O 65516,c1(C(N(CCNC(C(CC#C)C)=O)CC)=O)n[nH]c2ccc(F)cc12 65517,N1(C(c2cn(C)nc2)=O)C(C(=O)NC2CC(=O)NC2=O)CCC12CC2 65518,N1(C(=O)C=Cc2ccoc2)CCC2C(CCN2CC(O)CCl)C1 65519,C1(CC(N2CCCC(CCNC(=O)CC3OCCCO3)C2)=O)CN2CCN1CC2 65520,C1(C(N2CCCC(NC(C3C(c4n(C)ncc4)C3)=O)C2)=O)CCS(=O)(=O)CC1 65521,Cc1cc(C(=O)NC(C2CCOC2)CNC(c2cc(CO)n(C)n2)=O)ccn1 65522,C(C)(CO)(C(=O)NCCNC(C1CCCOC1c1cc(C(F)(F)F)n[nH]1)=O)OC 65523,Cc1cc(C)c(C#N)c(NCCc2csc(C)n2)n1 65524,C12CC(=NO1)C(=O)N1CCC(C(=O)O)(CC1)N(c1ccccc1)C2.CC(O)(C(=O)O)c1ccsc1.c1ccccc1 65525,CCC(C(=O)N(C(C)CN(C)C(c1cnn(CC)c1)=O)C)N(C)C 65526,Cc1sncc1C(=O)NCCCNC(C1CC1(C)C)=O 65527,N1(C(c2c(C)scc2)=O)CC(NC(=O)C#CC2CCCCC2)C2CCCCC12 65528,C1(C(=O)NCC(C)OC)(OC)CCN(C(c2ccc(Br)cc2F)=O)CC1 65529,c1(CCC(=O)OC2C(OC)CCC2)cnc2n1CCCC2 65530,CC1C(NC(c2nn(C(F)F)cc2Cl)=O)CCCN1C(=O)C(C)CC1CC1 65531,S(=O)(=O)(CC(=O)N1CCC(C)C1CNC(c1cccc(NS(N)(=O)=O)n1)=O)NC 65532,c1(C(=O)NCC(CC(C)C)NC(=O)C2=C(Cl)CCC2)ccc2c(c1)CCCC2=O 65533,c1(C(=O)NC2CC(C)(CNC(C3CCN(CC)C3)=O)C2)cc2cncn2c(O)n1 65534,N1(C(C(N2CCOCC2)C)=O)CCCC(O)(CNC(=O)C2=CSCCO2)C1 65535,CC1CC(CNC(=O)CCn2ccnn2)CN(C(=O)CC2(N3CCCC3)CC2)C1 65536,CC(C)C(CCN(C(=O)CC1COC(=O)C1)C)N=c1nc(-c2ccccc2)[nH]s1 65537,N1(C(CCC(C)OC(F)F)=O)CC2(CCCN2C(c2sccc2OC)=O)C1 65538,c1(CSC)nsc(N(C)C(C2CCC(F)C2)=O)n1 65539,c1(CC)nc(C)c(C(N2CCCCC2CNC(c2cnn(C)c2Cl)=O)=O)c(C)n1 65540,N1(C(c2csc(Br)n2)C(=O)NCCCSC)CCCCC1C(C)C(=O)OC 65541,C(=O)(C(O)(C(F)(F)F)c1cn[nH]c1)N1C(COC)CN(C(=O)CCCSC)CC1 65542,N1(CC(=O)NC(C2CCOC2)CNC(C(C)(C)C2CC2)=O)Cc2ccccc2C1 65543,N1(C(C(C2(O)CN(C(C(C)(CO)OC)=O)C2)F)=O)CCN(C)CC1C 65544,n1(CC)cc(NC(C2(CNC(C3C4CC5C(C4)C35)=O)CC3(CC3)C2)=O)c(C)n1 65545,N1(CC)CC(C(=O)NC(CCC2CC2)C(=O)NCC2(CC3CC3)CCC2)CC1=O 65546,N1(C(c2c(C)nn(CC)c2C)=O)CC(NC(c2n[nH]c(C)c2C)=O)C2(CCC2)C1 65547,Cn1cc(-c2cn(CCC(=O)N(C)C)nn2)cn1.C12CC1C(=O)NC2 65548,N1(C(c2cc(C)sc2C)=O)CCC(CNC(=O)CCOCCN(C)C)C12CC2 65549,C1(CCC)CN(C(=O)Cn2cc(Cl)cn2)CCN1C(=O)CN1CCC(C)(C)C1 65550,CCC(CC)C(F)C(=O)NC1CC2CCC1CN2C(C1CN2CCN1CC2)=O 65551,N1(C(C=C(C)c2ccccc2F)=O)CCCCC2(CCN(C(C3CCO3)=O)C2)C1 65552,c1(C(N2C3CC(NC(c4c(Cl)cn(C)n4)=O)(C3)C2)=O)n[nH]c2c1COCC2 65553,CC1=NOC2(CCN(c3cc(C(F)F)nc(Cl)n3)CC2)C1 65554,C1(NC(CC=C)=O)(CNC(c2ccc(C(=O)OC)nc2)=O)CCCCC1C 65555,c1(CC(=CC(=O)Nc2cn(C(c3ccccc3)OC)nc2)C)cc(Cl)ccc1Cl 65556,c1(N2C(C(=O)Nc3cnc(C(F)(F)F)nc3)CC(C)C2)ncc2[nH]ncc2n1 65557,C(=O)(C#Cc1ccc(Cl)cc1)NC1CN(Cc2cccc(C)c2F)CC1F 65558,C=CCCN=C(NCC1CCC(C(N)=O)O1)NCC1(F)CCC(C(=O)OC)CC1 65559,C1(NC(c2cnc(C3CC3)nc2)=O)CCCCC12CCN(C(=O)C=CI)C2 65560,c1(CC(=O)N(CCCNC(C2C(CC)OCC2)=O)C)ccc(O)cn1 65561,C=CCC(CC(C)C)C(=O)NC1COCC1CNC(=O)CCCn1cncn1 65562,C(=O)(CC1=CCCC1)N1CC(C(C)NC(C2(C(F)(F)F)CCCCO2)=O)OCC1 65563,C1(CNC(C2N(CC#C)CCC2)=O)CN(C(c2cc(COC)on2)=O)CCN1C 65564,c1(C(=O)O)ccnc(C(F)(F)F)c1.n12cc(nn1)C(C1CC1)C1(CCCC1)C2 65565,N1(C(C(CCC)OC)=O)C2CCC1CN(Cc1nc(C(C)OC)no1)CC2 65566,N1(C(c2cc(C)sc2)=O)C2CCC(C(=O)NCc3cncc(Cl)c3)C1CC2 65567,c1(C(N2CCCC(NC(C(CC)(C)O)=O)C2)=O)ccc(NC(C)=O)c(Cl)c1 65568,CC1CC(NC(=O)CCP(C)(C)=O)CN(C(=O)COc2ccc(Cl)nc2)C1 65569,N1(C(C(C)C(F)(F)F)=O)CCN2CCOCC2(CNC(=O)Cc2ccco2)C1 65570,c1(C(=O)NCC(C)NC(c2nnc(CN(C)C)s2)=O)ccccc1C1CC1(F)F 65571,N1(C(c2c(C)ccnc2O)=O)CC2(CCCC2NC(=O)CSC2CC2)C1 65572,CC(C)C(C)(C)C(=O)NC1CCCC(NC(C2(C)CC3CCC2O3)=O)C1 65573,Cc1ncccc1CCC(=O)NCC1(O)CCN(C(C2CCCC2)=O)C1 65574,CON1CC(NC(=O)N(CCC(=O)OC(C)(C)C)C)CC1=O 65575,CON(CCC(=O)N1CCC2CC2C1)C(=O)Cc1ncoc1C 65576,C1(NC(CN(C2CC2)CC)=O)CC2CN(C(c3nc(OC)c(C)s3)=O)CC2C1 65577,C1(NC(C2C(CC)C2)=O)CCCC1NC(=O)CC(=O)NCC(F)(F)F 65578,O=C1NCc2cc(C(=O)Nc3onc4ccccc34)ccc21 65579,c1(OC)cccc(C(C(=O)NC2CC(NC(c3sc(C)cc3Cl)=O)C2)OC)c1 65580,N1(C(C(C)NC(C(C)NC(=O)NC)=O)=O)CC(S(C)(=N)=O)C1 65581,c1(NC(=O)NCC2(OC)CCN(C(C)(C)C)C2)cc2ccc(C)cc2s1 65582,c1(-c2ccc(F)cn2)ccc(NCc2cnco2)c(F)c1F 65583,C(=O)(C1=NN2CCCN=C2N1)N1CCC(C2CC2)(C(=O)O)C1 65584,c1(OC)ccc(C=CC(=O)NC2(C3CN(C(=O)C(C)O)C3)CC2)c(OC)c1 65585,C(CC(=O)NCC1CC(SC)C1)N(C(=O)CC1CC1(C)C)CC 65586,c1(C(=O)NC2(C)CCN(C(C(C)Cn3cccn3)=O)C2)cncc(S(C)(=O)=O)c1 65587,CC(C)C(C(C)NC(=O)CCCCC1CC1)NC(=O)C(C)(F)F 65588,Cc1cc(O)ncc1C(N1CC(C2CC2)(C(=O)N(C)CC2CCCCC2O)C1)=O 65589,Cc1ccc(C(=O)NC2CC(O)CN(C(c3ccc[n+]([O-])c3)=O)C2)c(N)c1 65590,C1(NC(CC2(OC)CCOCC2)=O)CCC2(CC1)CN(C(=O)C(C(C)C)SC)C2 65591,c1(C(C)C)nc(NCCC2CC(F)C2)cc(=NC2CCN(c3cccs3)CC2)[nH]1 65592,N#Cc1ccc(C(O)C(=O)NC2CC(NC(=O)C(F)=CCCF)C2)cc1 65593,N1(C(C2(C(N)=O)CC2)=O)CC2CC2(CNC(=O)Cc2nccs2)C1 65594,C1(C(=O)Nc2cccc(NC(C(CC)(C)CC)=O)c2)CC2CCCCN2C1 65595,C1(NC(C23CC(COC)(OC2)C3)=O)CN(C(=O)CN2CCCC2)CC1N=[N+]=[N-] 65596,C1(NC(c2c(C)coc2)=O)CCCC1(C)CNC(c1ccoc1Cl)=O 65597,c1(CC(=O)NC2CC(N(C(c3c[nH]c(=NC)o3)=O)C)C2)c(OC)cccc1Cl 65598,C1(NC(C(C)c2ccsc2)=O)CC2CCC1N2C(=O)COc1ccc(F)cn1 65599,C1(C(=O)NCC(CN(C(CC2(C(=O)OC)CC2)=O)C)O)CNC(=O)CC12CCC2 65600,N1(C(CC(=O)OC)=O)CCC(C2CC2NC(c2cc(Br)n(C)c2)=O)CC1 65601,C#CC1(O)CCCN(C(=O)COCCNC(c2ccsc2)=O)C1 65602,C(=O)(C#CC1CCCCO1)NCC1(CCNC(CC(CC=C)(C)C)=O)CC1 65603,CC1(C)C(CNC(=O)C(=O)NCC2(C)COC(=O)N2)CCS1(=O)=O 65604,[N-]=[N+]=NCCC(=O)NC(C(=O)NCC(F)Br)C1CC1 65605,Cc1cnncc1C(N1CC(C(C)(C)O)(CNC(C2(C)CCCCO2)=O)C1)=O 65606,Cc1ccc(C(N2CC(N(C)C(c3ncn4c3CCCC4)=O)C2)=O)c2c1CCC2 65607,c1(C(N2CCC(NC(c3n(C)c(S)nn3)=O)CC2)=O)cccc(F)c1O 65608,C(CC(=O)NOCC1CC1)(c1ccccc1)NC(C1(CC)CCCO1)=O 65609,N1(C(C(CNC(=O)CC=Cc2ccccc2)O)=O)CCCC2C(O)CC12 65610,C1(C(=O)NCC=C(C)C)CCN(C(=O)CSC(C)(C)C)C12CCC2 65611,N1(C(C2(C)CC2)=O)CC2(CC2)CC1CNC(C1CC2(CCC2O)C1)=O 65612,Cc1cc(C(=O)NC(CO)C(C)NC(=O)C(O)Cc2ccccn2)c(Cl)cn1 65613,c1(CNC(c2ccn(CCC(F)(F)F)n2)=O)csc(CNC(C2CCOC2)=O)n1 65614,C=CCC(CC=C)C(=O)NCC1CCCN(C(C2(OC)CS(=O)(=O)C2)=O)CC1 65615,C(=O)(C1CCCc2nncn21)N1CCN(CCNC(C2(C)CC=CCC2)=O)CC1 65616,N1(C(C(COC)(F)F)=O)CCN2C(=O)C(NC(c3cnn(CCO)c3)=O)CC2C1 65617,O=C1CC(CC(=O)Nc2ncc(C3COC3)s2)c2ccccc2N1 65618,c1(C(C(=O)NCC(CNC(CNS(CC)(=O)=O)=O)C)=O)ccccc1 65619,C(=O)(CC1=CCOCC1)NC1CN(C(CCOCCCOC)=O)C1 65620,c1(C(=O)NC2CC(CNC(C(C=CCCC)O)=O)C2)cccc2nccn12 65621,C(c1cnc2ccccc2n1)=CC(=O)NC(C)(CNC(c1ccnnc1)=O)CO 65622,c1(CN2CCC(CC(=O)NCCC(=O)OCC)CC2)cc(C(F)(F)F)cc(Cl)c1F 65623,CCC(=O)CCC(=O)N1CCOCC1CCNC(=O)CCc1cccc(C)c1 65624,C1(C(N2CCC(CN=[N+]=[N-])C2)=O)(SC)CN(C(=O)CCC2CC(C)C2)C1 65625,Cc1ccc(C(N2CCC3CCCC23CNC(c2csnn2)=O)=O)c(=O)n1C 65626,CC1CN(C)CC(C(=O)NCC(C2CC2)N(C)C(c2nccnc2N)=O)O1 65627,c1(CC)n[nH]c(=NCC(C)(C)NC(c2cnc(O)c([N+](=O)[O-])c2)=O)s1 65628,Cc1ncsc1C=CC(N1CCC(N(C(=O)C(C)CF)C)C1)=O 65629,N1(c2ccc(N(C)C(c3ncncc3Cl)=O)cc2)CCc2ccccc2C1 65630,Fc1ccc(-n2nc(CSC3CCCCC3)nc2-c2cscc2Cl)cc1 65631,N1(C(CC(C)OC)=O)CC(C2(NC(=O)Cc3ccc(Cl)cc3C(F)(F)F)CC2)C1 65632,S(=O)(=O)(c1c[nH]c2ncc(Br)cc12)N(c1ccccc1)CC1(C)CCN(C)C1=O 65633,Cc1ccc2nc(C(=O)NCC3CCCC3NC(=O)COCCO)ccc2c1 65634,N1(S(C(C)C)(=O)=O)CCN(C(C2CCN(C(=O)C(C)(C)n3cccn3)C2)=O)CC1 65635,N1(C(CSc2c(C)cccc2)=O)CC2(CCN(C(=O)C=CC(C)C)CC2C(=O)O)C1 65636,C1(C(=O)NCCN(C(=O)COC)CCC)C2CCC1(c1ccco1)C2 65637,C(=O)(C(C)(F)C(=O)N1CCCC(CNC(c2nc(OC)ccc2C)=O)C1)OC 65638,CS(=O)(=O)C1(C(=O)NCC2(CCNC(C3CC(N=[N+]=[N-])C3)=O)CC2)CC1 65639,c1(CNC(C(N2C(C)CCOC2)c2ccccc2)=O)cccc(Cl)c1F 65640,C(=O)(C(C)(C)C)NCC(=O)NCCOCCNC(C1C(CC)C1)=O 65641,N1(C(c2cc(F)ccc2Br)C(=O)NCCCSC)CCN(C)C2(CC2)C1 65642,N1(C(C(=CC2CCCC2)C)=O)CCOCC(NC(=O)C=C(C)C)C1 65643,C(C1=NOC2CCCCC12)n1cc(C2(O)CN(C(CC3CC(=C)C3)=O)C2)nn1 65644,C1(NC(c2c(C)n[nH]c2)=O)CCCCCN(C(=O)C(O)C(C)(C)C)C1 65645,c1(C(N2C(CNC(=O)Cc3cncnc3)CC2)=O)ccc2c(c1)NCCC2 65646,C1(C(=O)NC(CC)C(C)O)CC(C)CN1C(C1CCCC(C)C1)=O 65647,Cc1n[nH]c(C)c1CC(N1CCC(NC(C2(n3cnnn3)CC2)=O)CC1)=O 65648,N1(C(c2cc(C)nn2C)=O)CCCN(C(C2CCCN(C(=O)OC(C)C)C2)=O)CC1 65649,CCCC(C(O)C(=O)N1CCC1C(C)O)NC(c1c(F)cncc1F)=O 65650,N12CCCC(C1)C2=O.c1(SCC(=O)N(CCNC(N)=O)CC)nnnn1C 65651,N1(C(C2NCCN(C(c3scc(C)c3C)=O)C2)=O)CCCC(C)(O)C1 65652,N1(C(C(=O)NCc2ccc(-c3ccc(Cl)cc3)cc2F)=O)CCC2CCC(C1)O2 65653,C(=O)(C1=CC2(CCOCC2)C1)NCCC1(O)CCN(C(C(CC)(C)F)=O)C1 65654,c1(C(N2CCC(F)(C(N(C)C3CC3)=O)CC2)=O)c(Cl)ccc(Cl)c1F 65655,c1(C(c2nnnn2CCCSC)NCC(=O)NCCC)cccc(OC)c1F 65656,N1(CCC)CC(C(=O)N(C(C)CN(C(=O)CCc2cccnc2Cl)C)C)CC1=O 65657,Cn1ccnc1C(CF)NC(=O)C(N)Cc1ccoc1 65658,C(=O)(C(C)CC(F)(F)F)NC(CC(C)C)CNC(=O)C1=CCSC1 65659,N#Cc1c(F)cc(NC(N2CCN(c3ncccn3)CC2)=O)cc1Br 65660,CC1C(NC(=O)CNS(=O)(=O)N(C)C)CCCN1C(=O)CNC=O 65661,CC1CC(CNc2ccccc2COCC(N)=O)CCN1CC(N)=O 65662,C1(C(N(CC#C)CCF)=O)(CC=C)CN(C(=O)CC2CCC(C)C2)C1.C 65663,CON1CC(C(=O)NC(C(N2CCC(C)(CCO)C2)=O)c2ccco2)CC1=O 65664,C(=O)(C(CC#CC)NC(c1coc(CC)n1)=O)N1CCC(OCC=C)CC1 65665,c1(CCC(=O)NC2CN(C(C3C(C(=O)OC(C)(C)C)C3)=O)C2)ccccc1Br 65666,N1(C(CN(C)C(=O)C2CC2)=O)CCCCC(NC(C2CCCCC23CC3)=O)C1 65667,c1(C(N(CC(C)(C)NC(CC(C(=C)C)OCC)=O)C)=O)c(Cl)ccc(F)c1C 65668,C1(NC(Cc2n(C)ncc2)=O)CC12CCN(C(c1ccc(Br)cn1)=O)CC2 65669,C#Cc1cccc(CC(=O)NC(C(=O)NC(C)C(=O)OCC)c2ccco2)c1 65670,n1(CC(N2C(CNC(C(C)OCC=C)=O)CC2)=O)nnc(C2CC2)n1 65671,Cc1ccc(C=CC(=O)NCC23CCCC2CCN3C(=O)COC(C)C)cc1C 65672,C1(CNC(c2c(C#C)c[nH]n2)=O)CC2CN(C(=O)C(O)C(C)C)CC12 65673,c1(C(N(C(C)CNC(c2cc(O)nc(O)c2)=O)C)=O)ccc(F)c2ccncc12 65674,Cc1cc(Cl)c(Br)cc1S(=O)(=O)NCC1(CN)CCCCCC1 65675,c1(C(=O)NCC(CNC(=O)C(F)(F)c2nccs2)OC)cccc(F)c1N 65676,c1(NC(C(=O)NCCC2CN(C)C(=O)C2)=O)cccc2c1COCC2 65677,CC1CCCC1CC(=O)NCC(C)(F)CNC(=O)Cc1cccs1 65678,C(CS(=O)(=O)CC(=O)NCC(C)(CNC(c1c(C)ncn1O)=O)OC)OC 65679,C(=O)(CCCCSCC)NC(C(=O)OCC)C1CN(C(C2(C(N)=O)CC2)=O)C1 65680,c1(C(=O)OC(CC(=O)NC)OCC)cc(C)n(-c2ccc(Cl)cc2)c1C.OCC 65681,c1(OC)ccc(C(C)C(=O)NCCCCCNC(=O)CSC2CC2)c(C)c1 65682,c1(C(N2CCN(CC3CN(C(=O)CCC4CC4)C3)CC2)=O)ccc2nc[nH]c2n1 65683,C(=O)(C(C)(C)CCC#N)N1CC(C(N(c2ccc(F)cc2)C)=O)C2(C1)CC2 65684,c1(C(N(C(C)CNC(=O)C=Cc2ccnn2C)CC)=O)ccc(C(C)C)cn1 65685,C1(C(C)NC(C(C)(C)NC(=O)NCC=C)=O)CCCN(C(c2cc(Cl)c[nH]2)=O)C1 65686,CCC(CC(=O)NC1CC2CCC1CC2NC(c1cn(C)[nH]c1=N)=O)C(C)C 65687,Fc1c(I)c(SCC2COCc3ccccc32)nc2ccc(Cl)nc12 65688,c1(-c2cccc(NC(C3N(CC)CCCC3)=O)c2)cnn2c1NCCC2 65689,CN1CCC(F)(CNC(=O)C(CCC2CCC2)NC(=O)CCc2csnn2)C1 65690,CC1OCCCC1C(=O)NC(C)(C)CN(C(=O)Cc1nnn(C(C)(C)C)n1)C 65691,C1(O)(CCNC(C2CCS2(=O)=O)=O)CCN(C(=O)Cc2ccsc2)C1 65692,Nc1ccc(-c2nc(C(N3CCCC3)=O)n(-c3ccnc(Br)c3)n2)nc1 65693,CCCC(C(=O)NC1CC2(CCCN(C(=O)C(C)(C)F)C2)C1)S(N)(=O)=O 65694,c1(CC(=O)NC23CC(CNC(C(CCC)OC)=O)(OC2)C3)ccc(CO)c(C)c1 65695,C=CCCCCCCCC(=O)NC(C1CCN(C(=O)CCC(=C)C)C1)(C)C 65696,c1(C(=O)NC(CSCC)C(=O)NC2CCN(N(C)C)CC2)cccc2nncn12 65697,C1(NC(=O)NC2(CO)CC2)(Nc2cccc(-c3cnco3)c2)CCCCC1 65698,N1(CCN(CCCOC)C)CCC(=O)N(Cc2ccc(F)cc2C)C1=O 65699,C1(N2C(=O)CN2CCC(=O)OC)CCS1(=O)=O.C1(CC2CC2)CCCO1 65700,CN1CCc2[nH]nc(C(=O)NCC3CC3CNC(=O)C3=C(Cl)CCC3)c2C1 65701,c1(OCC(=O)N(CCNC(C2(C(C)C)CCC2)=O)CC)ccc(Br)cc1 65702,N1(C(=O)CC2CC3(CCC3)CO2)CC2CN(C(C34CCC(CC3)CO4)=O)CC2C1 65703,N1(C(C(C(C)C)C#N)=O)CCc2nc(CNC(=O)CCn3ccnn3)sc2C1 65704,c1(C(=O)NCC2CCCC2O)cnn(-c2cccc(Cl)c2)c1C(F)F 65705,Cn1cnc2[nH]c(C(=O)NC3CC(NC(=O)CC4CC5COCC45)C3)cc12 65706,C1(NC(C)=O)CCN(C(C2COCC2NC(=O)C(=CC2CCCC2)C)=O)C1 65707,c1(N(C)Cc2nc(CC)sc2)cc(C)c(S(=O)(=O)N2CCCC(C)CC2)cn1 65708,C1(C(=O)NCCC2CCOC2)CC2(CC2)CN1C(=O)C=CC(F)F 65709,C=CCC(C)(C)CC(c1nnnn1CCSC)NC1CC(C)C1 65710,Cc1nnc(N(CC(=O)OCc2ccc(CCC(F)(F)F)cc2)C)n1C 65711,N1(C(CS(CCC)(=O)=O)=O)CCC2CCN(C(C3CCCSC3)=O)C2C1 65712,c1(C(=O)NCCCOCCNC(C=CC(CC)C)=O)cn(C)nc1Cl 65713,C1(Cc2cn(CCC=C)nn2)CCCCN1C(c1scnc1C(C)(C)C)=O 65714,c1(C(N2CC3C(N(C(=O)CCCSC(C)(C)C)C)C3C2)=O)ccc2ncccn12 65715,N1(C(C(C2CCCC2)NC(CCCCC)=O)=O)CC2(CCC(=O)NC2)C1 65716,c1(C(N2C3CN(C(Cn4c(C)ccc4C)=O)CC2CC3)=O)c(Cl)c([N+](=O)[O-])nn1C 65717,CC1=NOC(C(=O)NC(CNC(C2CC(NS(C)(=O)=O)C2)=O)CC(C)C)C1C 65718,N1(C(c2c(C)nc(COC)s2)=O)CCC(C2CC2)C1CNC(C1CC1C(C)O)=O 65719,c1(CCC(=O)NCC(CN(C(c2nc(CCC)sc2)=O)C)O)nnc(S)nc1O 65720,n1(CC(=O)NC(CN(C(C(C)N(C(C)=O)C)=O)C)(C)C)nnc2ccccc12 65721,N1(C(c2cnc(OC)s2)=O)CCCCC1CCNC(=O)CCc1cc(Cl)cs1 65722,c1(C(=O)NC2CC3(CN(C(C(C(C)C)C)=O)C3)C2)ccc2c(c1F)CCC2 65723,CCC(C)(C#N)C(=O)N1CCC(NC(c2cc(Cl)ccc2OC(C)C)=O)CC1 65724,c1(-c2ccc(C)c(OC(F)F)c2)ccccc1S(=O)(=O)NCC(O)CO 65725,N1(C(C(N2CCN(C)CC2)C)=O)CC(NC(C23CCCN2CCC3)=O)CCC1C 65726,N1(C(=O)C(F)CC2CCOC2)C(CNC(CCO)C2CCC2)CCC1SC1CC1 65727,C1(C(=O)N(C2(CN3CCCC3)CN(CC)C2)C(c2cc(C)cs2)=O)CC(C)OC1C 65728,c1(COC)cc(C(=O)NCC(c2cccc(C)c2)NC(C2CC2(F)F)=O)c(C)o1 65729,C1(C(=O)NCC(C(CC)C)(C)O)CC(C)(C)CCN1C(=O)Cn1nccn1 65730,c1(C(N2CC(C)(NC(=O)C=CCN3CCCC3)C2)=O)ccc(F)c(Br)c1F 65731,C1(C)(C(N2CC(N(C(=O)CCCC3CC3)C)C(O)C2)=O)CCC2(CC1)OCCO2 65732,c1(OC)nn(C)c(Br)c1C(=O)NC1CC1NC(C1(C)CC1(F)F)=O 65733,C(CC(=O)N1CC2(CSC2)C1)(C(F)(F)F)NC(=O)C=CC1CCOC1 65734,Nc1cc(F)cnc1C(=O)NC(CCOCCO)C(=O)NCC(O)C(F)F 65735,c1(C(N(CCCN(C(=O)Cc2ccc(F)c(Cl)c2)C)C)=O)nc2cnccc2s1 65736,CN=c1[nH]c(C(=O)NCC2CCCCN2C(c2cn(C)cn2)=O)cs1 65737,N1(C(CC2N(CC)CCC2)=O)CC2(CC(NC(=O)CC34COCC(C3)C4)CO2)C1 65738,Cc1cc(Br)c(F)cc1C(=O)NC1CC(C(=O)NC(C2CCOC2)C)C1 65739,C1(OCC)CC2(C1)CC2C(N1CC(OC)C1)=O.N12CCC1C(=O)NCC(=O)C2 65740,C#CC1(C(N2CCOCCC2C)=O)CCN(C(=O)CCC(C)(F)F)CC1 65741,CC1CCCC(CC(=O)NC(C2CCN(C(c3ccn(CCF)n3)=O)CC2)C)O1 65742,c1(C(=O)NCC(c2ccccc2)CNC(CSC)=O)cc(C2(O)COC2)on1 65743,C(C(CNC(c1cc2n(n1)CCC2)=O)C(F)(F)F)NC(CSCCOC)=O 65744,C1(F)(CNC(C(C)(C)OC(C)=O)=O)CCN(C(=O)C(C)C(C)(C)C)CC1 65745,C1(C(=O)NC(CC(C)C)CO)CC12CCN(C1CCC(=O)N(C3CC3)C1=O)CC2 65746,CN=c1cc(C(=O)NC2CC(C)N(C(C3CCC(OC)CC3)=O)C2)cc[nH]1 65747,N1(C(=O)CCc2cccnc2)CC2(C1)CN(C(C1(CCO)CC1)=O)CCO2 65748,c1(C(c2nnnn2C2CC2)NC(C=C)C2CCC2)cn(C)nc1C(F)F 65749,CCC(C(=O)Nc1cccc(C(C)(C)C)n1)C(C)C 65750,C1(C(N2CCN(C(=O)Nc3ccc(F)cc3F)CC2)=O)CCc2cncn2C1 65751,Cc1ccc(C(=O)N(C(=O)CSc2nncn2C2CC2)Cc2ccncc2)cc1 65752,C1(NC(C=CC(C)(C)SC)=O)COCCC1NC(=O)C(C)(O)C1CC1 65753,c1(C(=O)NC2(CCOC)CCN(C(=O)C3=CCCO3)C2)cc(Cl)ccc1C 65754,C1(CN(C(C2C(C)C2C)=O)C)CCN(C(C2(c3ccccc3)CCCO2)=O)CC1 65755,C1(CNC(c2ccc(Br)o2)=O)CCC2(CN(C(c3c(O)cccc3F)=O)C2)O1 65756,CC1CCCC1C(N1CC(C)(CNCc2ccc(Cl)s2)C1)=O 65757,C1(C(N2CC(C(=O)NC3CCCC(SC)C3)(COC)C2)=O)CCCS(=O)(=O)C1 65758,Cc1ncncc1C(=O)NC(C1CC=CCC1)C(=O)N(C1CCN(C2CC2)C1)C 65759,C1(N(C(=O)CC2CCC2)CCC)CCN(C(=O)CCc2ccn(C)n2)CC1 65760,C(=O)(C(C)=NOCC#N)NC(COC)C(=O)NCC(O)(COC)CO 65761,N1(Cc2cn(C)nc2I)CC(=O)N(CCc2ccn(-c3ccc(Cl)cc3)n2)C1=O 65762,N1(C(CC(=O)NCC)=O)CCCC1(C)C(=O)NC(C1(OC)CCC1)C 65763,Cc1cc(=O)oc(C)c1C(=O)NCCc1ocnc1CNC(=O)C=CC1CCC1 65764,C1(F)(C(N2CCC(C)(CCNC(C3(C#C)CCC3)=O)C2)=O)CCCN(C)C1 65765,c1(C(=O)NCCCN(C(=O)C(C)(O)C2CCOC2)CC)scnc1Cl 65766,c1(C(=O)NCc2cccc(CNC(C3(CC)CC3)=O)c2)cnc(Cl)cc1Cl 65767,CCCC(CCC)C(=O)N1CCC(C(=O)NC(C)CC(C)C(F)F)O1 65768,C1(CCNC(C2CC(=O)NC2)=O)CCCCN1C(=O)C(=O)Nc1ccccc1 65769,c1(OCCC(=O)NCC(C)CN(C)C(C2CC(F)C(=O)N2)=O)cccc(Cl)c1 65770,c1(NC(=O)OCC2C(C(=O)OC(C)(C)C)C2)ccc(F)c(C=O)c1 65771,N1(C(C(N2CCN(C)CC2)C)=O)CCC(C2CCCN(C(C3(CF)CC3)=O)C2)C1 65772,C(CC(F)F)(C(=O)NCCN1CCCCC1C)NC(CC=C)=O 65773,c1(C(=O)NCC(CCOC)NC(c2oc(C)nc2C)=O)ccc(C(C)C)nc1O 65774,N1(C(c2nnc(C)o2)C)CCC(NC(c2cccc(F)c2Cl)=O)C(C)C1 65775,C(CNC(c1cncnc1)=O)(CC(F)(F)F)NC(c1cnc(SC)s1)=O 65776,C=CC(C)(CC)C(=O)NCc1ccc(CNC(=O)C(C)NC(=O)CC)cc1 65777,n1(CC)cc(Br)c(C(=O)Nc2ccccc2-c2cccc(C(F)(F)F)c2)n1 65778,c1(C(N2CC(CNC(C3C4CCCCCC34)=O)OCC2)=O)cccc2c1COC2 65779,c1(C(=O)NCC2(NC(C3CC(C)OC3)=O)CCCCC2)cc2n(c1)CCSC2 65780,C1(NC(c2cccc(C)c2)=O)CC2(C1)CN(Cc1cc(O)ncc1Br)C2 65781,C(=O)(C(CC)C(C)(C)CC)NC(CN(C(C(C)OCCC=C)=O)CC)CC 65782,C1(CC)CN(C(=O)Cc2occc2C)CC1NC(c1ccc(SC)cc1)=O 65783,C12CCN(C1)C(=O)CO2.c1(OCCNC(C2CC(=C3CCC3)C2)=O)cccnc1 65784,Cc1c(C(=O)NC2(C(=O)NC3COCCN(C)C3)CC2C)cncc1F 65785,CCC(C)CC(C)C(=O)NCC(C(C)C)NC(c1n[nH]c(C)c1Cl)=O 65786,c1(C(=O)NC2CCC(N(C(C(CC)n3ccnc3)=O)C)C2)ccc(F)c(C)c1O 65787,Cc1cnc2n1CC(C(=O)NCC(C)N(C)C(c1csc(Br)c1)=O)CC2 65788,C(=O)(CCP(C)(C)=O)NCC(C1CCCN1C(=O)C(F)(F)c1ccnn1C)(C)C 65789,c1(NC2C(C)C2)ccc(Cl)c(C(=O)OCC2CCCO2)c1.N12CC(C1)CC2=O 65790,c1(N(C(c2ccc(Br)cn2)C(=O)NC2COC2)C)cccc(Br)c1F 65791,C(=O)(CCC(O)C(C)(C)C)NCC(C)CNC(c1csc(=N)[nH]1)=O 65792,Cc1cc(C(=O)N(CCC(C(C)(C)C)NC(=O)CCC2CC2(F)F)C)cc(C)n1 65793,N1(C(c2c(C)con2)=O)CCC2(CCCN2C(=O)C=CBr)C1 65794,N1(C(c2cc(CC)nnc2C)=O)CCCC12CCN(C(c1cc(Cl)c(Cl)[nH]1)=O)C2 65795,Cc1nnnn1CC(=O)NC1(C)CC(NC2(C)CN(C(=O)OC(C)(C)C)C2)C1 65796,c1(C(N(C2CCN(C(C3(CO)CCC3)=O)CC2)CCCC)=O)nnc(O)nc1O 65797,CC1CCCC1NC(=O)C#CCNC(=O)COCc1nc[nH]n1 65798,Cc1cc(NCN2CCN(c3ccc(C(F)(F)F)cn3)C3CC23)cc(C#N)c1 65799,c1(C(N(C(CNC(C2(C(=O)OC)CC2C)=O)C2CC2)C)=O)ccc(F)cn1 65800,C(c1ccc(C)c(Cl)c1)=CC(=O)NCC1CN(C(CC(=O)NCC)=O)CC1(F)F 65801,Cc1cccc(CC(N2CCCC(NC(=O)C(F)n3ccnc3)C2)=O)c1Cl 65802,C(=O)(C(CCC)CC(C)C)N1CC(NC(C2(CC#C)CCCCO2)=O)C(C)C1 65803,C(=O)(C1CCCc2n[nH]cc21)N1CCC(COC)(NC(c2c(C)ncn2O)=O)C1 65804,C1(c2ccc(OC)cc2)C(C(=O)OC)=C(C2CCOCC2)N(C)C(=O)N1C 65805,c1(C(=O)NC(c2ccccc2)C(C)NC(C(C)=C2CC2)=O)ccc(Cl)c(C)c1Cl 65806,CC(N=c1[nH]c(=NC2CN(C3CCC3)C2)[nH]c2c1CCCC2)c1cn(C)nn1 65807,N1(C(C2(OC)CCCC2)=O)CCC(NC(=O)C(C)CC(F)F)C2(CCC2)C1 65808,CCC(CC(F)(F)F)N=c1nc(N2CCC(F)(C#N)C2)c2c([nH]1)CCC(C)C2 65809,N1(C(C=C(C)C(C)C)=O)CCC(CCNC(c2cccn2C)=O)CC1C 65810,N1(C(C(C(C)C)(C)O)=O)CCC2(CCCN(C(=O)CCn3cc(Cl)cn3)C2)CC1 65811,C1(F)(CNC(C(OC)OC)=O)CC(CNC(=O)Cn2cc(C3(O)COC3)nn2)C1 65812,Cc1nn2cc(C(N3CCCC3CCNC(=O)C(C)N3CCC3)=O)nc2s1 65813,c1(OCC)c(C(=O)NCCCCCNC(C2(C)CC3CCC2C3)=O)cccc1F 65814,Cc1cc(N)ccc1C(N1CCCC(N(C)C(C2CN(C3CCC3)C2)=O)CC1)=O 65815,C(C1=NOC2OCCC12)OC(C1CS(=O)(=O)CC1N1CCOCC1)=O 65816,n1(CC(=O)NCC2(OC)CN(C(=O)CC3NC(=O)NC3=O)C2)c(C)c(C)sc1=O 65817,c1(C(N2CCC(NC(c3c(CC)ocn3)=O)C(C)C2)=O)nccn2cc(C)nc12 65818,c1(NC(C2CC(=C)C2)=O)cnc(OC)cc1C(=O)Nc1cnc(Cl)c(C(F)F)c1 65819,c1(OC)ncc(C(N2CCC(C(=O)Nc3cnc(Br)c(Cl)c3)C(O)C2)=O)cc1Br 65820,N1(C(C2C(C(C)O)C2)=O)CCCC1CNC(=O)CCn1cc(Cl)cn1 65821,c1(C([N+]2([O-])C(C)CN(C(C3CC3C#N)=O)CCC2)=O)ccc2nnn(O)c2c1 65822,c1(C(N2C(C(N(CCCC)CCO)=O)CC3CC32)=O)ccc([N+](=O)[O-])cc1O 65823,c1(CC)cc(N2CC3CC3(CN(C(c3ccccc3CO)=O)CC)C2)nc(C)n1 65824,C(C)(CC(=O)N1CC=CC1C(=O)NCCCc1nc(C)no1)SC 65825,C1(CNC(C(C2(O)CCC2)NC(C(C)NC(=O)OC)=O)=O)CNC(=O)C1 65826,Cc1cc(C(N2CCOCC2CC2CCCN(C(=O)C(C)C)C2)=O)cn(C)c1=O 65827,c1(C(=O)NCC2(C)CC(NC(c3c(CC)onc3)=O)C2)[nH]c(O)nc1C 65828,CCCC(C(=O)NCC1(C)CCCN1C(c1ncoc1C)=O)OCC 65829,N1(C(C(c2ccoc2)NC(=O)CC(C2CC2)C2CC2)=O)C2C=CCC1CC2 65830,c1(CN(C2CCCC(O)C2)C)cc(Cl)cnc1O 65831,C1(CC(C2(F)CCCCC2)NCc2n(CCC3(C)CC3)nnn2)CCC(C)CC1 65832,N1(C(C(C)(C)O)=O)CCCC2CN(C(c3cnc4sccn4c3=O)=O)CCC12 65833,C12(N(C)C)CCC(C(=O)NCCC(C)(C)NC(=O)Cc3cnnn3C)(CC1)CC2 65834,C1(C(N2CC(N(C)C(C3(C)CCOC3)=O)C2)=O)CCCCC(C)(C)C1 65835,c1(C(=O)NCC2N(C(c3nn(CC)c(O)c3)=O)CC2)cc[nH]c2nccc1-2 65836,C1(F)(CNC(c2cc(Cl)c[nH]2)=O)CN(C(C2CCCSC2)=O)C1 65837,c1(C(=O)NC2(C)CN(C(C3OCCOC3(C)C)=O)C2)ccc(F)c(F)c1 65838,CCC(CC(=O)NCC1CN(C(=O)C(c2cnn(C)c2)=O)C(C)(C)C1)C(C)(C)C 65839,c1(C(=O)OC)cnc(C(=O)NCC2CC3(CCO2)CC3)c(N)c1 65840,C1(CC)CC(CC(=O)OCc2ccccc2-n2cccn2)CCO1 65841,c1(C(=O)NC(C2CCCN2C(c2cn(C)nn2)=O)C)nc(Br)c[nH]1 65842,C(C(C)CC(=O)NC1CC(NC(=O)C=Cc2ccc(-c3ccccc3)o2)C1)OC 65843,C(=O)(CS(=O)(=O)Cc1cccs1)NCC(C)NC(c1nncs1)=O 65844,C1(C(=O)NC2(C)CCOC2)C2CN(C(=O)CCc3nc[nH]n3)CC12 65845,c1(C(=O)NCC(C)NC(C2(Cl)C3CCC(=O)C23)=O)cc[n+]([O-])cc1 65846,C1(CNC(CC(C)SC)=O)CC(F)(F)CN1C(=O)C=C(C)C1CC1 65847,CC(c1ccc(F)cc1)=CC(=O)N(C(C)CCNC(=O)C(C)(C)CO)C 65848,C1(NC(C2(C)C(C)C2)=O)CCC12CCN(C(c1ccc3nn(C)cc3c1)=O)CC2 65849,N1(C(c2nc(C)nc(O)c2)=O)CCC2(CCCN(C(=O)CC3(O)CCOC3)C2)C1 65850,N1(C(c2cc(OC)n(C)n2)=O)CC(NC(=O)Cc2sccc2Cl)C2CCCC2C1 65851,c1(OC)cc(=O)n(C)cc1C(N1CC(N(C(=O)C(O)Cn2cncn2)C)C1)=O 65852,N1(C(C2(Br)C(C)(C)C2)=O)CCCCC12CC(NC(c1cccc(C3CC3)c1)=O)C2 65853,CCC(C)CCCCC(=O)NCCC1(CNC(=O)C(C)CC(F)F)CC1 65854,C1(N(c2ncncc2F)Cc2c(C(=O)OCC)c[nH]n2)CCC2(CC1)CNC2 65855,c1(C(N2CC(Cn3cc(-c4ccc(Cl)c(F)c4)nn3)C2)=O)cc2n(n1)CCCC2 65856,c1(OC)c(C(=O)NCC2(NC(C3(C)CCOC3)=O)CCC2)ccc(Cl)c1Cl 65857,C1(CNC(CN(CC)CC)=O)CC2CCC1N2C(c1cc(F)ccc1OC)=O 65858,C1(CNC(c2cnn(C(F)F)c2)=O)CCN(c2ncnc(Cl)c2F)CCC1(F)F 65859,N1(C(c2scc(C)c2)=O)CC2(CC2)CC1C(=O)NCc1c(Cl)cccc1Cl 65860,C12(NC(C=Cc3c(C)cccn3)=O)CCCN(C(=O)C=CC3CCOC3)CC1C2 65861,C(=O)(CCCCC(C)=O)N1CCCC(C)(C(=O)NC(CCC)(C)CC)C1 65862,CC(C)(C(=O)N1CC2CC1C2NC(=O)CCCCn1ccnn1)C(N)=O 65863,C1(N)CCOC1C(N)=O.C(=O)(C(C)CO)N(CC(O)C(C)C)CC=C(C)C 65864,c1(C(N(CCCCN(C)C(c2cnnn2C2CC2)=O)C)=O)ccc([N+](=O)[O-])n1C 65865,Cc1ocnc1C(N1CCCC1CC(=O)N(C1CC(O)C1)C)=O 65866,N1(C(c2n(CCCC)ncc2)=O)CCC(NC(=O)C=CC(C)C)C(O)C1 65867,C(F)(F)(C(F)(F)F)OCC(=O)N(C)CC1(NC(Cc2ccc(C)o2)=O)CC1 65868,C1(N(C(C2(CC=C)CCOC2)=O)C)CCN(C(=O)C(Br)=C(C)C)CC1 65869,Cc1cscc1C(=O)N(C)CCOCCN(C(=O)CCc1nnc(C2CC2)o1)C 65870,c1(-c2nc(C(c3c(OC)cccc3)C)on2)cc(C)cc(O)c1 65871,C1(C(=O)N(CC)Cc2nccs2)(CC)CCCN(C(=O)C=Cc2ccccc2)C1 65872,N1(C(c2nnn(CC)c2C)=O)CCC(C2CC(NC(C3(CC)CCC3)=O)C2)CC1 65873,CC1CC(C)CN(C(=O)CC2CCN(C(=O)CCc3nc[nH]n3)CC2)C1 65874,c1(C(N2CCC(NC(CCCC=C)=O)C2C2CC2)=O)ncc(P(C)(C)=O)cn1 65875,CCC(C)C(=O)N(C(C)CCNC(c1ccn(C2CCC2)n1)=O)C 65876,c1(CCC)ccccc1C(N1CCCC1c1cn(Cc2ccco2)nn1)=O 65877,CCCC(CCNC(=O)C(C)N(C(c1cncc(OC)c1)=O)C1CC1)C1CC1 65878,C1(NC(C(=O)NCC)=O)CC2CCC1N(C(C1(N(C)C)CCCC1)=O)C2 65879,N1(CCC)CCCC(C(N2CCC(CNC(=O)CSc3c(C)n[nH]c3C)C2)=O)C1 65880,C1(NC(=O)CCN2CCCC2)C2CC(CN(C(=O)CSC(F)F)C2)C1CO 65881,C1(C(=O)NCC(C(=O)NC2(CC)CCCCC2)O)CC(=O)CC12CCC2 65882,N1(C(c2c(COC)nn[nH]2)=O)CCN(C(=O)Cc2n[nH]c(C)n2)CC1C(C)C 65883,c1(C(=O)NCC2(C)CCN(C(CC(C)n3cccc3)=O)C2)n[nH]c2c1CSCC2 65884,CN1CCN(C(c2ccccc2CC#N)=O)CC1CNC(=O)C(C)(C)C(N)=O 65885,c1(C(CNC(c2nnn(-c3ccccc3)n2)=O)NC(C(C=C)O)=O)ccc(C)cc1 65886,C(=O)(C(O)CC(C)C)NCCCN(CCC)C(c1c(C(=O)NCC)cccc1)=O 65887,N1(C(C23C(C)OC(CC2)C3)=O)CC2(CC(NC(=O)CCS(C)(=O)=O)CO2)C1 65888,C(CCC(C)C)(C(=O)NCCN1CCCCC1=O)NC(CC(CCC)C)=O 65889,N1(C(c2cn(CC)nn2)=O)CCC2(CNC(C3CCCC3O)=O)CCCCC12 65890,C1(NC(CC2(C=C)CCOCC2)=O)CN(C(c2cnc(C)o2)=O)CC2(CCC2)C1 65891,C12(C(N3C(CC(=O)NC(C(C(=O)OC)C)C)COCC3)=O)CCC(C1)OC2C 65892,C1(NC(COCC(c2ccccc2)C)=O)CCC2CC1CN2C(=O)Cn1cnnc1 65893,C1(C(=O)NC(CNC(c2ncnc(C)c2C)=O)(C)C)CC12CCc1ccccc12 65894,C1(C(F)F)(CNC(c2scc(OC)c2)=O)CCN(C(C2CN(C(C)C)C2)=O)C1 65895,C(=O)(CCC(C)(C)[N+](=O)[O-])NCC1(C)CC(NC(c2c(C)onc2C2CC2)=O)C1 65896,CC(C(=O)NC1CCN(C(c2[nH]cc3c2CCC3)=O)CC1)C(F)(F)C(F)F 65897,CC1CC2=C(C(=O)N1)C(c1sccc1S(C)(=O)=O)NC(=S)N2C1CC1C 65898,N1(C(c2ccc(CCC)cc2)=O)CCN(C(C2C(C)(C)C2(F)F)=O)CCC1C 65899,C=CCC(C)(C)CC(=O)NCCN(C(=O)CC1CCC(=O)NC1)C1CC1 65900,C1(NC(=O)C=CC2CCCCC2)CCCCN(C(=O)Cc2ccc(Cl)cc2Cl)C1 65901,C1(NC(C2CCC(CC(=O)NCC3CCCSC3)C2)=O)CCC2(CC2)C1 65902,c1(C(N2CCN(C(CS(CC)=O)=O)CC(O)C2)=O)ccc2nnc(O)n2c1 65903,C1(C(N2CC(CC=C)(NC(=O)COCC(F)(F)F)C2)=O)CCc2nncn2C1 65904,c1(C(=O)NC2(CCCNC(Cn3ncc(CC)c3)=O)CC2)ccc(N)cn1 65905,C12(C(N(CC(F)Cl)C)=O)CCCC1CCN2C(c1n[nH]c2c1CCC2)=O 65906,C1(NC(=O)CCCc2ccccc2)CC12CCN(C(=O)CCC1OCCO1)CC2 65907,CCCS(=O)(=O)C(C)C(=O)NCCNC(c1ccc(Br)c(OC)c1)=O 65908,c1(C(=O)NC(CNC(C(C)SCC)=O)C2CC2)c(C)cnnc1O 65909,c1ccc(C2CCN(CCNC(N3CCCC3)=O)C2)nc1 65910,CCC(C(C)(C)O)NC(=O)C(C1CN(C(=O)CCC(=O)NC)C1)OC 65911,CC1(C)CCC(CNC(c2cc(CNC(c3n[nH]cc3Cl)=O)on2)=O)C1 65912,C1(C(=O)NC(C#C)CC2CC2)CCCCC1NC(C1(C2CC2)CC1)=O 65913,O=S(=O)(c1ccc2nc(O)oc2c1)C1CC1.C12=CNC(=NCc3cccnc31)S2 65914,C(=O)(C(C)(C)CC(C)(C)C)NC1CN(C(C(CC)CC(F)F)=O)CC(C)C1 65915,N1(CC=CC(=O)NC(C)CN(C)C(C2(C)CC2Br)=O)CCOCC1 65916,C12(NC(=O)CSc3ccncc3)CC(C1)N(C(c1cccnc1O)=O)C2 65917,N1(C(c2ccc(C)c(C)c2)=O)CC2CC(NC(C3CC(C)(C)C3)=O)CC1C2 65918,C1(C(N(C2CCC(O)CC2)C)=O)COCCC1NC(C1(C#N)CCOS1)=O 65919,C1(COC)(CNC(C2CC(C(C)C)C2)=O)CCN(C(=O)C(c2ccc(Cl)s2)=O)C1 65920,C(=O)(CCC(C)NC(=O)C(c1cncnc1)C)NCC1(CC)CCOC1 65921,c1(C(=O)NCC2N(C(CS(CC)=O)=O)CC(O)C2O)cc(OC)cc([N+](=O)[O-])c1 65922,c1(N2CCC(N(C(C=C(CC)CC)=O)C)CC2)cc(C)nc2nc(C)nn12 65923,N1(C(C(C)O)=O)CC(CNC(=O)C(=O)Nc2ccc(Br)cc2)C2(CCC2)C1 65924,Cc1cc(C(=O)NCC(O)CNC(C2NC(=O)OC2C)=O)ccc1C1CC1 65925,N1(CC(N2CC3C(N(C(=O)CCn4ccnn4)C)C3C2)=O)CCc2sccc2C1 65926,N1(C(C(C2CC2)OCC)=O)CCC(C)(NC(=O)CCC2CC2C)CC1 65927,C1(CC=C)(NC(=O)Cc2cnn(C(F)F)c2)CCN(C(=O)CN2CCOC2=O)C1 65928,C(=O)(CCC(C)(C)C)NC(C1(O)CCN(C(Cn2c(C)csc2=O)=O)C1)C 65929,N1(C(c2n(CC)ncc2Cl)=O)CC2CCC2(NC(=O)CCc2cnn(C)n2)C1 65930,c1(C(N(CCOC)CCNC(C23CCCC2CC3)=O)=O)nn(C)c(C)c1Br 65931,c1(C(=O)NCC2(NC(C(C)Sc3ccccc3Cl)=O)CCC2)cnc2n1CCC2 65932,c1(CN2CCC(NC(c3c(C)nc(OC)s3)=O)C(F)C2)ccc([N+](=O)[O-])cn1 65933,Cc1ccc(C)n1CC(N1CC(CCNC(C2CC(=O)N(CC(C)C)C2)=O)C1)=O 65934,CCC(C)(COC)C(=O)NC(C)CCCNC(c1ccn(COC)n1)=O 65935,C1(C(=O)NC(C2CCCN2C(c2cnc(O)s2)=O)C)CS(=O)(=O)C1 65936,C1(C)(OC)CCCN(C(=NCCF)NCC(C)(O)C(F)(F)F)C1 65937,Cc1cc2c(CC(=O)NC3CC(NC(c4cc(C(=O)OC)sn4)=O)C3)csc2s1 65938,C=CCC(CC(=O)NCCCF)NC(c1coc(N(C)C)n1)=O 65939,C12(NC(C(C)c3cccs3)=O)CCCC1N(C(c1ccc3n[nH]cc3n1)=O)CC2 65940,C1(CC(=O)N(CC(CNC(C2C(c3ccc(C)s3)C2)=O)(C)C)C)CCC(=O)NC1 65941,N1(C(c2ccc(C#C)o2)=O)CCC(F)CC1C(=O)NCCc1ccncn1 65942,C1(C(=O)NC2C(NC(c3ncnc(C)c3C)=O)CC2)Cc2cccc(F)c2O1 65943,c1(C(N(C)CC2COCCN2C(C2CC23CCC3)=O)=O)cc2c(nn1)CCCO2 65944,c1(C(N(CCN(C(=O)CC2C=CCCC2)C)C)=O)nn(C(C)(C)C)cc1Br 65945,c1(C(=O)NC2(CC=C)CN(C(=O)CNS(C)(=O)=O)C2)cc(NCC)ccc1C 65946,CC1=C(C(=O)NCC2CC3COCC3N2C(=O)CC(C)CC(C)C)CCS1(=O)=O 65947,c1(C(=O)NC2CC(CCNC(=O)CC(=O)Nc3nccs3)C2)cc([N+](=O)[O-])c[nH]1 65948,C(N=c1[nH]c(=NCCN2CC=CCC2)c2ccccc2[nH]1)c1cc(C)c(Cl)cc1 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65967,C(C)(C(C)C(=O)N1CCOC(C)C1)NC(C1(C(C)C)CCC1)=O 65968,c1(C(N(C2CCN(C(=O)CC3CCNC3=O)C2)CCC)=O)ccc(CC2CC2)s1 65969,c1(C(N2CCC(C(C)NC(c3ncccn3)=O)C2)=O)sc2sccc2c1Cl 65970,C(=O)(CCCCCCCCC1CC1)N1CCCC(NC(C(C)CC(N)=O)=O)CC1 65971,C#CCCCCC(=O)NCC(CC1CC1)C(=O)N(CCCCC=C)C 65972,N1(C(C23C(CN(C(c4c(CC)noc4)=O)C2)C3)=O)CCC(C#N)CC12CC2 65973,C1(C2(O)CN(C(c3cc(C)nc(N(C)C)n3)=O)C2)(CNC(CC)=O)CC1 65974,N1(C(c2c(C(C)C)onc2)=O)CC(C)CN(C(=O)C(O)CN(C)C)C(C)C1 65975,C(=O)(C1CCCc2ncccc21)N1CCC(N(C(CC)=O)CCO)CC1 65976,C1(CNC(C(c2cccnc2)NC(C2C(C(=O)OC)C=C2)=O)=O)CC(=O)N(C)C1 65977,N1(C(C2CC(CNC(C(C(C)C)=O)=O)C2)=O)CCN(C)C(CO)C1 65978,c1(NC(c2nc(CC)c(C)s2)c2nnnn2CC2CC2)cnn2c1C(=O)NCC2 65979,Cc1ccn2cc(C(=O)NC(C3CCCN3C(c3c[nH]c(Br)c3)=O)(C)C)nc2c1 65980,C(=O)(CCCCCC(C)C)N(CCOC)CCNC(=O)C#CC1CCOC1 65981,C(CS(C)(=O)=O)N(C)C(C1CCC1NC(=O)CCC1CC1)=O 65982,c1(C(=O)NC(C)CCCNC(=O)C=Cc2ccco2)cccc(Br)c1 65983,CCC1=NOC(C(N2CCCC(N(CCF)C(c3cn(C)cn3)=O)C2)=O)C1 65984,N1(C(c2c(C)nn(C(C)C)c2)=O)CCC(CNC(=O)COC2(C)CCC2)C(C)C1 65985,c1(OC)cc(C(=O)N(C)CCN(C)C(c2cc(N)ccn2)=O)cc2cnn(C)c12 65986,c1(CN2CCC(CC(=O)NCc3cc(O)cc(Br)c3)C2)ccc2c(c1)C(=O)CC2 65987,CONC(=O)CNC(C1(F)CN(C(=O)C(=C2CCCCC2)F)C1)=O 65988,C1(C(=O)NC2CN(C(CCC(=C)C)=O)CC2(C)C)CC2CCCC(C1)C2 65989,CC(C)CC(=O)C(=O)NC1CCCC(C(=O)NCCC2(O)CCOC2)C1 65990,c1(C(N(CC(=O)N(CC2CC(=C)C2)C(C)C)C)=O)n[nH]c2c1COC2 65991,C1(CNC(c2n(CC)ccn2)=O)CN(C(=O)C(C#N)C(C)C)CCN1C 65992,CC1CC(NC(c2nccnc2Cl)=O)CN(Cc2ncccc2C(F)(F)F)C1 65993,CCC(CC)C(C)C(=O)NCC1CCCN1C(=O)CNC(c1cccc(C)c1)=O 65994,CC(C)C(C(=O)NC(C)(CO)C1CCC1)N(C)C 65995,c1(SC)cc(C(=O)NC(C)C(C)NC(c2conc2-c2ccccc2)=O)c(C)o1 65996,Cc1ccc2nc(C(=O)NCc3ccc(C(F)F)cn3)[nH]c2c1 65997,CC(C)(CNC(=O)CNc1cccnc1)CC(=O)NCC(C)(O)C1(C)CC1 65998,C(C(C)N=c1cc(Cl)nc(SC)[nH]1)SC.S1(=O)(=O)CCC(=O)N1C 65999,c1(C(N2CCC(CNC(c3cc(C)on3)=O)C2)=O)cc2ccccc2c(O)n1 66000,C1(OC)CN(C(=O)CC2CCN(C)CC2)CC1NC(=O)CN1CSCCSC1 66001,c1(CN2CCC(C(=O)NCCSCC)C2)cccc(Br)c1Br 66002,CN1CC=CCC1CC(N1CC(N(C(=O)Cc2ccsc2)C)C(O)C1)=O 66003,C1(C)(CNC(C2(SC)CC(=O)C2)=O)CN(C(c2cc(Cl)n(C)n2)=O)CC1C 66004,c1(C(C(=O)NC2CC(C(=O)OC)C2)N(C(C#C)C)C)csc(CC)n1 66005,C(C(C(C)(C)C)NC(=O)Cc1cc(C)on1)NC(Cc1ccc(C)o1)=O 66006,CCC(C)C(O)C(=O)N1CCCN(C(c2cc(Br)c(C)cn2)=O)CC1 66007,CCCCCCC(CC)C(=O)N1CCCC12CCN(C(c1cc(Br)n[nH]1)=O)C2 66008,N1(C(C2CCC(OC)CC2)=O)CC(NC(C2CCOC(C)(C)C2)=O)C(C)(C)C1 66009,N1(C(c2cc(OCC)n[nH]2)=O)CC2(CCN2C(C2CCC(=O)C(C)C2)=O)C1 66010,Cc1[nH]cc(C(N2CC(O)(CN(C)C(C3(O)CC4CCC3C4)=O)C2)=O)c(=O)c1Cl 66011,CC1=NS(=O)(=O)NC=C1C(=O)N1CC2CC1C2CNC(=O)CC(O)C(C)C 66012,C(=O)(CC(C)(O)COC)NCC(CNC(C=CC(CC)=CC)=O)OC 66013,N1(C(c2c(C)c(C(F)(F)F)n[nH]2)=O)CCN(C(=O)C(Cl)=CCl)C(C)C1C 66014,CC(CC(=O)N1CC2CCC1CC2NC(C1(C)CCCCO1)=O)P(C)(C)=O 66015,c1(NC(C2C(C(=O)OC)C2)=O)ccc(I)c(C(c2cc(F)ccc2Br)OC)c1 66016,C(=O)(C(C)(O)C(F)(F)F)N1CC(NC(c2c(OCCOC)cccc2)=O)C(C)C1 66017,C1(C(=O)NC2CC3(C(C(N4CC(NC(N)=O)C4)=O)C3)C2)CCCCC(=O)C1 66018,CC1CC(CNC(c2cnn(CCF)c2)=O)CN1C(c1cccnc1O)=O 66019,n1(CCCC)ncc(C(=O)N(CCC)CCNC(=O)CC(C)N(C)C)c1C 66020,CCC(O)C(C)C(=O)NCCCN(C1CCCC1)C(c1cnc(C2CC2)[nH]1)=O 66021,N1(C(c2c(SC)c(F)ccc2)=O)CCCC1C1CCCN1C(=O)C(F)F 66022,N1(C(Cn2cc(-c3cccc(CC)c3)nn2)=O)CCC2(CC1)OCCO2 66023,c1(C(=O)NCC(C)CNC(=O)CC2(C)CCC2)cn(C2CCN(C)C2)nn1 66024,c1(OC)cnc(F)c(C(=O)N(C(=O)C(c2cc(F)cc(F)c2)OC)CCC#N)c1 66025,N1(C(CC(C(=O)OC)C)=O)CCC(C)(C)CC1C(=O)NCC1NC(=O)OC1(C)C 66026,c1(C(N2CCC(NC(=O)Nc3cccc(C)c3)C2)=O)c(Cl)ccc(O)c1Cl 66027,C1(NC(C2ON=C(C)C2)=O)(CNC(c2cncc(F)c2Cl)=O)CC2CCC1CC2 66028,c1(NC(C2N(C(C(CSC)O)=O)CC(F)C2)=O)ccc(O)cc1C 66029,Cc1cc(CCC(N2CC(NC(C3CCS3(=O)=O)=O)CC2C)=O)cc(C)c1 66030,C(=O)(CC(O)C(C)C)NCC(Cc1cn(CCN(CC)CC)nn1)(C)C 66031,N1(C(C2CC(=C)C2)=O)CCC(C)C1CNC(c1cnc(C2CC2)nc1)=O 66032,Cc1ccc(CC(=O)NCC(CC(C)C)NC(C2(C3CC3)CC2)=O)cc1C 66033,c1(C(=O)NC2CCCN(C(c3cccnc3Cl)=O)C2)ccc2nnc(Br)n2c1 66034,N1(C(CSCCC)=O)CCN(C(c2cn(CCC)nc2C)=O)CC(O)C1 66035,C1(NC(CN(C(=O)CSCCOC)CC)=O)COCC1N(C)C 66036,C(=O)(C(C)(F)C(=O)N1CCC(=CCNC(c2ccc(CO)c(C)c2)=O)CC1)OC 66037,CC(C)C1=CCC(NC(C2(NC(=O)C=CC3CC3)CCN(C)C2)=O)CC1 66038,C(=O)(CC(C)(C)c1ccc(C)cc1)N(C(CNC(C(C)=CC)=O)C)C 66039,C1(CNC(CCCC(C)O)=O)CC2(CO1)CN(C(=O)C(F)(F)CO)C2 66040,C(=O)(CCC(C)(C)F)N(CCCNC(=O)CC1CCCC1(F)F)C 66041,n1(CC)ncc(CNC(=O)CCN2CCN(C(=O)C(C)NC(C)=O)CC2)c1C 66042,N1(Cc2cnc(OCC)c(Cl)c2)CCC2C1CCCN2c1nccc(N(C)C)n1 66043,N1(C(C2C(OC)CC2)=O)CC(NC(c2ccc(Cl)c(F)c2N)=O)C2(CCC2)C1 66044,N1(C(C(N2CCOCC2)C)=O)CCCCC(N(C(=O)C=C(C2CC2)C2CC2)C)C1 66045,CC1CC(C(=O)NCC2C3CN(C(c4ccc(Cl)nn4)=O)CC23)CCC1C 66046,N1(C(C(C)OCC=C)=O)CCN(C(c2ccc(SC)s2)=O)CC1CC 66047,C1(C#N)(C(=O)NCC2(OC)CN(C(c3cncc(C(C)C)c3)=O)C2)CCSCC1 66048,C1(OC)CC2C1CCN2C(C1(NC(=O)Cc2ccn(C)n2)CC1C)=O 66049,C(=O)(C(c1ccoc1)NC(=O)C(C)N(CCSC)CC)NCC(=C)C 66050,NS(=O)(=O)N1CCCC(C(=O)NCC(O)CNC(c2c[nH]c(C(N)=O)c2)=O)C1 66051,c1(NC)scnc1C(=O)NCCCC(C)NC(=O)Cc1csc(C(C)OC)n1 66052,CCCCCCCCCCCNC(C1C(NC(c2cc(C)ns2)=O)C1)=O 66053,Cc1ccccc1C=CC(=O)NC(C)CCN(C)C(C1CC2CC2C1)=O 66054,c1(C(N2CCC(NC(CN(CC)CC)=O)C(O)C2)=O)cccc2c1OCCO2 66055,c1(SC)cc(C)c(C(N2CC(CNC(C3(C)CCOC3C)=O)C(O)C2)=O)o1 66056,CC1N(C(=O)C(Cc2ccoc2)NC(c2cccnn2)=O)CCOC1(C)C 66057,CCCCC(C(=O)NCC(CC(N1CC(CO)CC(C)(C)C1)=O)OC)C(C)C 66058,C(C)(CC(=O)NCC(C)(C)CNC(c1cc(N)c(F)cc1F)=O)(C(F)F)N(C)C 66059,C1(CNC(CCOC)=O)CC2(CCOCC2)CN1C(=O)CC1CC2CCC1C2 66060,C1(NC(CCC2(C)CC2)=O)CCC(O)CN(C(c2c[nH]c3ccccc23)=O)C1 66061,n1(CC(C)C(=O)NC2CC(F)(CNC(=O)CC3(C)CC3)C2)ncc2c1CCCC2 66062,C1(CNC(=O)Nc2ccc(Br)cn2)CCCC(CF)C1 66063,CC1(C)CN(C(=O)C(O)CNC(c2cc3cccnc3[nH]2)=O)C2CCCC12 66064,N1(C(c2c(C)ncs2)=O)CCC2(CC1)CCN(C(c1csc(C)c1C)=O)C2 66065,c1(C(C)N(CC(C)C#N)C(=O)CN(C)C)ccc(Cl)s1 66066,Cn1cnc(S(N)(=O)=O)c1C(=O)NC1CC(CNC(c2cncn2C)=O)C1 66067,C=CCC(CC(F)F)C(=O)N1CC(CNC(=O)COCc2cccs2)CC1(C)C 66068,C12(C(=O)NC3C(C)CN(C(C4(n5cnnn5)CC4)=O)C3)CC3CC(C(=O)N1)C2C3 66069,c1(C(CC(=O)OC)=O)ccc(F)cc1[N+](=O)[O-].C1CCC(=O)O1 66070,C1(=O)NNc2nccnc2N1.C1(CNC(=O)OC(C)(C)C)CC2CCC1O2 66071,c1(NCCCCNC(C(CC)OC)=O)ncccc1C 66072,Cc1cccc(C)c1C(=O)NCCC1COCCN1C(C1CC1C)=O 66073,C1(C(N2CCC(O)(CNC(COCC#C)=O)C2)=O)CCc2nnn(C)c2C1 66074,c1(C(=O)NC2C(C)(C)CCN(C(C(C=C=C)C)=O)C2)cc(C)cc2c1OCC2 66075,C#CCC(C)(CC)C(=O)NC1COCCC1C(N1CCC1(C)C)=O 66076,CCC(CC(=O)N1CCC(CCNC(=O)C(C)(C)CF)C1)c1ccc(OC)cc1 66077,c1(C(=O)NC2CCCN(C(C(C)OCCCC)=O)CC2)nc2c(s1)COCC2 66078,c1(CCC(=O)NC2CC2CNC(C2(F)C3CCCC23)=O)ccc2ncccc2c1 66079,CC1(C)CCOC(Cn2nnnc2N2CCC(C3CC(C(N)=O)CCO3)CC2)C1 66080,O=C(CCC1CC1C(F)(F)F)NCC1CC1NC(=O)CC1CCC1 66081,c1(C(=O)NCC2(F)CCN(C(C3CC(OCC)C3)=O)C2)ccc(C)c(C)c1 66082,C12(C(=O)NCC3CCC(NC(C(C)(C)C(N)=O)=O)CC3)CCCCC1OCC2 66083,C1(NC(CNC(C)=O)=O)(CNC(c2nccn2C)=O)CCC(C)CC1 66084,C(CC(O)CO)NC(C1C=CCN1C(C12CCCC1C2)=O)=O 66085,C1(NC(=O)CCCCN2CCCC2)CC(F)(F)CC1C(=O)O 66086,C1(CNC(Cn2cnc(CC)n2)=O)CN(C(=O)COC2CC=CC2)CC1C 66087,C1(NC(C(C)(C)CF)=O)CCN(C(=O)C(C2(O)CCCCC2)(C)C)CC1CO 66088,c1(C(N(C)CC2CCCCN2C(=O)CC2(CO)CC2)=O)cnc2ccccc2n1 66089,C1(CC)CN(C(=O)Cc2nc(Cl)cs2)CCN1C(c1csc(C)n1)=O 66090,C(CCOCC)(C(=O)N(C)CCN1CCCC1)NC(C(CC)n1ccnc1)=O 66091,c1(OC)cc(CO)ccc1C(N1CCCC(C)C1CNC(=O)CSC)=O 66092,Cc1cc(=O)oc(C)c1C(=O)NC1CS(=O)(=O)CC1NC(C1CCCC(=O)C1)=O 66093,C1(O)(CNC(C2CC(=C)C2)=O)CCCN(C(c2ccc(Br)c(C)c2)=O)C1 66094,c1(OCC)cc(C(=O)NC(CCN(C)C(C2(O)COC2)=O)C(C)(C)C)oc(=O)c1 66095,N1(C(c2c(C)n(CCO)cc2)=O)CCCC(NC(C2CC(C)(F)C2)=O)C1C 66096,c1(C(=O)NC2C(NC(c3cc(C)sn3)=O)CCC2)ccc2c(c1)CN(C)C2 66097,c1(C(N2CCC(NC(c3cncc(C(C)(F)F)c3)=O)CC2)=O)nnn2c1CCC2 66098,c1(CC(C(=O)N(C(CC#C)C)C)NC(=O)C(C)CC=C)cnn(C)c1O 66099,Cn1cc(C(=O)NC2C3CC(NC(=O)CCC4CCC4)CC23)ncc1=O 66100,c1(OCC)ncccc1CC(=O)NCC1CCN(C(C2(n3nccn3)CC2)=O)C1 66101,C(=O)(C1=CCCCC1C)NCC(C)(C1CC1)NC(c1occ(C)c1)=O 66102,Cc1nc(Cl)ccc1S(=O)(=O)NCC1CN(Cc2cccc(O)c2O)CCO1 66103,c1(-c2c(OCCC)ccc(F)c2)ccc2c(c1)CN(C(=O)C(C)=O)CC2 66104,Cc1cc(F)c(Cl)cc1C(=O)NCC(C)CN(C)C(c1ccc(C#N)nc1O)=O 66105,c1(C(=O)NCC(C(C)(C)C)NC(c2ncc(C)c(C)c2)=O)cc(C#N)c(C)cn1 66106,N1(C(C=CCC)=O)CCN(C(c2cnn(CC)c2CC)=O)C(C(C)C)C1 66107,c1(NC(C2(OC)CCC(C)CC2)c2nnnn2C)ccc2nn(C)c(C)c2c1 66108,C1(C(=O)NC2(C(=O)NCC3C4CC5C(C4)C35)CCOCC2)CCC2CC1CO2 66109,CN1CC(CC(N2CC(N(C)C(C3CC(=C4CCC4)C3)=O)C2)=O)C1 66110,C1(NC(CC(=O)NCC2CC2)=O)(CO)CCCN(C(C2CCCO2)=O)C1 66111,c1(OC)cc(C#N)ccc1CNC1CC1C(=O)NCC1CCO1 66112,C(=O)(C1CCc2snnc21)NC(C(C)NC(c1cnn(CCN(C)C)c1)=O)C 66113,c1(-c2nc(C)[nH]n2)nc(-c2cccc(OC(C)C)c2)nn1Cc1cncc(F)c1 66114,C1(CNC(CCc2nc(C)sc2)=O)CCCCN1C(C1(C)CCCC1)=O 66115,C1(O)(C(C)NC(C2(F)CCOC2)=O)CCN(C(=O)COCC2CCCO2)CC1 66116,Cn1cc(C(=O)NCC2CN(C(=O)Cc3ccsn3)CC(C)(C)C2)c(O)nc1=O 66117,C1(C(=O)NC(c2nn[nH]n2)CC)(C(C)C)CCN(C(C2CCS(=O)CC2)=O)C1 66118,N1(C(c2ncn(CC)c2)=O)CC2(C(=O)N(C)Cc3cnc(C)s3)CCC1CC2 66119,C=CC(C(=O)NC(Cc1ccco1)C(=O)N1CC(C)(CCO)C1)OC 66120,S(=O)(=O)(c1ccc(Br)s1)N(CCN1CC(C)CC(C)C1)C 66121,N(C(=NCCCOC)N1CCC(NS(C)(=O)=O)C1)C(C#C)C(C)C 66122,C12(NC(c3cc(COC)cn3C)=O)CCC(C1)N(C(=O)C(F)=CC1CC1)C2 66123,N1(C(c2cc(CC)oc2C)=O)CCN2CCN(C(c3cc(F)c[nH]3)=O)CC2C1 66124,CC(=O)CCC(=O)N(C(C)CNC(=O)CCNC(c1ccsc1)=O)C 66125,c1(NCC(=O)NC(C)(C)COCC(F)(F)F)ccc(F)cc1I 66126,Cc1ccsc1C=CC(N1CCC(C(C)NC(=O)CCC(C)C)C1)=O 66127,C(=O)(C(=O)N=S(C)(C)=O)N1CC(NC(CC2CCC(C)CC2)=O)C(C)CC1 66128,N1(C(c2n(C)ccc(=O)c2)=O)CCOC2(CCCCC2NC(C2CCOC2)=O)C1 66129,N1(C(C=C(C)C(C)C)=O)CCC(NC(c2cccc(N)c2F)=O)C(F)(F)CC1 66130,N1(C(C(C)=NCc2scc(CC)n2)=O)CC(NC(C)=O)C2(CCS(=O)(=O)CC2)C1 66131,N1(CC(C2CCOC2)F)CCC(NCC(F)F)CC1 66132,N1(CC)CCCC1CC(=O)NC(C)CNC(C1(C)CC1C)=O 66133,CC1CN(C(C2(O)CCSC2)=O)CC1CNC(c1cc(-c2cnn(C)c2)on1)=O 66134,c1(-n2cc(-c3ccn(C)n3)nn2)ccccc1NC1CN(c2ccc(F)cc2)C1 66135,N1(Cc2ccc(C)o2)CC(C(N2CC3CC2(C(F)(F)F)C3)=O)CCC1=O 66136,C1(C(=O)NC(CSC)(C)C(=O)NCC2(O)CCCC2)CC2C(C1)C2(F)F 66137,C1(N(C(=O)CC2CC=CCO2)CC)CCN(C(=O)C(=O)N(C)C)CC1 66138,c1(CC(C(=O)N(C(C)CNC(C2CC2F)=O)C)C)ccc([N+](=O)[O-])cc1 66139,Cc1cccc2[nH]cc(CC(=O)NC34CC3CN(C(=O)CC3CCCN3C)C4)c12 66140,C(=O)(C1=NOC(C)C1C)NC1(CC=CC(=O)NCC(CC)(C)OC)CCCCC1 66141,C1(NC(CSCC(C)C)=O)CCN(C(=O)CC(=O)NC2CC2)CC1O 66142,C1(C(=O)NC2(C)CCN(C(=O)Cc3n[nH]c(=N)s3)CC2)CSc2ccccc2O1 66143,c1(CC(=O)NCC(CNC(CC2(C)CC2)=O)O)ccc(C(N)=O)cc1 66144,N1(C(c2c(SC)ccs2)=O)CCN(C(=O)Cn2c(C)csc2=O)C(CC(F)F)C1 66145,c1(NCc2ccc(OC(C)C)c(F)c2)nccc(=NC(CF)CF)[nH]1 66146,CC(=O)CCN=C(NCc1cc2ccccc2o1)NCC1CN(C2CC2)C(=O)O1 66147,c1(NC(CN(C(C)C)C)C)nc(N2CCOC(CF)C2)nc2sccc12 66148,C#CCC(CC(F)F)C(=O)NCCC1CC(NC(=O)Cc2ccnn2C(C)C)C1 66149,O=C(C1c2c[nH]nc2CN1C(c1cnc(O)o1)=O)NC1C2COCC12 66150,c1(C(=O)NC2C(NC(c3coc(C(F)F)c3)=O)CCC2)ccc2c(c1)COC2=O 66151,C(=O)(C1=CCCSC1)NC1C(NC(CCc2ccc(OC(C)C)cc2)=O)CCC1 66152,C1(NC(c2ccnc(OCC3CC3)c2)=O)CCOCC1F 66153,CCC(C)CC(=O)NCC1CCC(NC(=O)C(C)(Cl)Cl)C1 66154,N1(C(CCCc2c(C)ccs2)=O)C(C(=O)NCCOC2CCC2)CC2CC12 66155,C#Cc1ccc(C(=O)NCC(C)N(C(c2ccc(OC)c(N)c2)=O)CC)cc1 66156,C12(NC(C(C(C)C)N(C)C)=O)CCC(CC1)N(C(C1CC3C=CC1C31CC1)=O)C2 66157,C1(CNC(c2ncn(C)n2)=O)CN(C(=O)C(C)(F)F)CCO1 66158,C1(C(=O)NC2CC(O)(CC3(C)COC3)C2)CCC(C#N)C1.n12cc(nn1)C2 66159,CCCCC(C)CCC(=O)NC1(CNC(=O)C(F)(F)C2CC2)CCCCC1 66160,C(=O)(C(F)CCC(C)(C)C)N(C1(C(N2CCC(C(=O)NC)C2C)=O)CC1)C 66161,C1(C(=O)NCCC2(C(NOCCOC)=O)CCC2)CCCC1C 66162,Cc1nnc(O)c(C(=O)NC2CN(Cc3cccs3)C2)c1C 66163,C1(C(=O)NCCC(C)NC(c2ncoc2Br)=O)CCCCCC1(F)F 66164,c1(C(=O)NC2(C(NOCCOCCOC)=O)CCCC2C)ncc(F)cc1N 66165,C1(CC#C)(C(N2CCCC(NC(=O)CCN3CCOCC3)C2)=O)CCOCC1 66166,N1(C(C(C=C)(C)CCOC)=O)CCOC2(CCN(C(c3cncnc3C)=O)C2)C1 66167,N1(C(C(CC)C)=O)CC2CC1CN(C(=O)C(N1CSCSC1)C)C2 66168,N1(C(CN(C(C)=O)C)=O)CCC(F)(C(=O)NC(CC2CCC2)CO)CC1 66169,N1(C(c2ccn(C)n2)=O)CCN(C(=O)C=CC(C)(C)C)CC1c1ccccc1Cl 66170,C1(NC(Cc2ccc(C)cc2)=O)CCN(C(c2cc(C)cnc2Cl)=O)CC1(C)C 66171,C1(C2(O)CCN(C(c3cscc3Cl)=O)CC2)(NC(=O)COCC2CCOC2)CC1 66172,C1(NC(c2cnc(Cl)s2)=O)CCCN(C(c2cnc3c(c2)COC3)=O)CC1F 66173,N1(C(C(C)=CC)=O)C2CCC1CN(C(=O)Cc1ccc(O)c(O)c1)C2 66174,c1(CC)ccnc(N(C)C(=S)NCC(c2ccc(F)cc2)O)c1 66175,N1(C(CC2C=NN(C)C2=O)=O)CC(NC(=O)CCn2ccccc2=O)CC(F)C1 66176,c1(N(C)C)c(F)cc(C(=O)NC2CC2C(=O)NCc2nc(Br)cs2)cc1F 66177,CCCCC(O)CC(=O)N1CC(C)(C)CC1CC(=O)N(C1CCCCCC1O)C 66178,N1(CC=CCNC(C=CCN(C)CC)=O)CCC(NC(c2sccc2Cl)=O)CC1 66179,c1(C(N2C(CN(C(C(CC)=O)=O)C)CCC2)=O)cc(SC)cc(CC)c1 66180,C(CCC(O)C(=O)NCC1CC(=C2CCC2)C1)NC(=O)C(F)F 66181,S(=O)(=O)(c1cccnc1NC(CO)C1CC1)NC(C(C)(C)C)c1ncccn1 66182,C1(NC(C2(C=C)CCC2)=O)CCCN(C(c2ocnc2-c2ccccc2)=O)C1 66183,C(C(C)(C)C#CC(=O)NC1(C(N)=O)CC1)NC(Cc1scc(C)c1)=O 66184,c1(C(N2CCC(CNC(C3(N(C)C)CC3)=O)C2)=O)cccc2c1CCCC2 66185,C(=O)(C(F)C1=CCCCC1)NCCN(C(C(Cc1c(C)cccc1)C)=O)C(C)C 66186,N1(C(c2c(CCC)[nH]cc2)=O)CC2CC1CN2C(C1CC1C(C)C)=O 66187,N1(C(C(C)(C)c2cnco2)=O)CC(NC(c2cnc(C(C)(C)C)o2)=O)C2(CC2)C1 66188,c1(SC)cc(C)ccc1C(N1CCN(C(C2CSC2)=O)CC1CS(C)(=O)=O)=O 66189,c1(C(N2C(C(=O)NCCSC)CCC2)=O)cccc(-c2cccs2)n1 66190,N1(C(CC2CCC(NC(=O)Cc3ccsn3)C2)=O)CC(CO)C(O)C1 66191,c1(NC(N2CCC(c3cc(=N)[nH][nH]3)C2)=O)nc2ncccc2o1 66192,c1(C(=O)NCc2c(C3CN(C(C(C=C)O)=O)C3)ocn2)ccc(C2CC2)cc1C 66193,Cc1n[nH]cc1C(=O)NC1CCC(NC(C2(CCCN(C)C)CCCC2)=O)C1 66194,CC(C)C(CCN(C(=O)CC(=O)NCCOC(C)(C)C)C)NC(=O)C(F)=CC1CC1 66195,c1(CC)nc(C#N)cc(=NCC2(NC(C3CCOC3C)=O)CCCC2)[nH]1 66196,Cc1nc(C)c(C(=O)NC2CCCC(NC(c3cnc[nH]c3=N)=O)C2)o1 66197,Cc1n[nH]c2nc(O)c(C(=O)NC3(CNC(=O)C=CC(F)(F)F)CCOC3)cc12 66198,N1(C(C2CCC(OC)CC2)=O)CC(F)(F)CCC1C.C(=O)(N)N 66199,N1(C(c2n(C)ccc2)=O)CC(O)C(O)C1CNC(C1CC(=C(F)F)C1)=O 66200,N1(C(C2(CC)CC2)=O)CCCC1C(C)NC(C)=O 66201,CC1(C)CN(C(=O)COc2ccc(F)c(F)c2)CC1NC(=O)CC1CC12CC2 66202,C1(N(C(c2cc(SC)oc2C)=O)C)CC2CCC(C1)N2C(=O)CCc1cnc[nH]1 66203,c1(C(=O)NCC(CNC(C(CC#C)O)=O)C)cnc(Br)c(O)c1 66204,c1(C(=O)NCCC2CCCN(C(=O)CC3CC(CF)C3)C2)ccc(CO)c(Cl)c1 66205,c1(C(N(CCCOCCNC(c2c(C)ocn2)=O)C)=O)sc2ccccc2c1Cl 66206,CC1C(NC(=O)CC(C)(C)C(F)F)C(C)CCN1C(=O)CCOCC(F)F 66207,CC1CC(N=c2[nH]c(=NCC3(c4ccccn4)CCC3)c3ncccc3[nH]2)CS1 66208,c1(C(N(C2CCCN(C(=O)C(O)C(F)F)CC2)CC)=O)nc(C)c(C)nc1C 66209,N1(Cc2ccc(C(=O)NCC)cc2)CC(C)OC(C)C1C 66210,N1(CC(=O)NC2CN(C(CCOCC#C)=O)C2)CCCC1C 66211,C1(NC(c2cccc(COC)c2)=O)CCN(C(c2cccc(CO)n2)=O)CC1O 66212,C1(CC)CN(C(C2(F)CC=CC2)=O)CCC1NC(C1CCC(CC#N)CC1)=O 66213,c1(NC(=O)C(N2CCCC(Cc3ccccc3)C2)=O)cc(Cl)cnc1Br 66214,C1(C(CC)C)CCCN(C(c2cncc(CNC(=O)C=CC3CCC3)c2)=O)C1 66215,C(N=c1[nH]c(=NCCCOCCCO)[nH]c2cc[nH]c12)c1nccc(C)n1 66216,C(C(O)CCNC(c1csc(-c2nc[nH]n2)n1)=O)NC(=O)CCc1cnn[nH]1 66217,c1(NC(C(N2CCC(NC(C3CCCCN3C)=O)CC2)C)=O)ccc(Br)cc1F 66218,C1(C(C)NC(=O)Cc2nnc(O)s2)CN(C(c2ccc(C(F)F)o2)=O)CCO1 66219,c1(C(=O)NC2C(NC(CCN(CC)CC)=O)CC2)cnc(O)cc1O 66220,c1(CC(=O)NC2CCC(CNC(Cc3ccn(C)n3)=O)C2)c(F)cccc1C#N 66221,Cc1ccnc(C(N2CCCC2(C)CNC(=O)C(N2CCCC(C)C2)=O)=O)n1 66222,C12(C(C)NC(C3CC(C)N3C(=O)C=Cc3ccnn3C)=O)CCC(CO1)C2 66223,N1(C(C(CCSC)(C)C)=O)CCC=C(C(=O)N(C)CC2C(C)(C)C2(C)C)C1 66224,c1(NC(C2CN(C(c3n(C)c(S)nn3)=O)CC2F)=O)cccc2c1CCO2 66225,C1(C(C)NC(C(C2CC2)OCC)=O)CCN(C(c2csc(CC(C)C)n2)=O)CC1 66226,CCC(C(=O)N(CCCNC(C1CCC(=O)NC1)=O)CCO)C(C)(C)CC 66227,c1(C(=O)NCC(CNC(C(C)n2cccn2)=O)CO)ccc(C#N)cn1 66228,c1(C(=O)NC2(CNC(C3CCNC(=O)C3)=O)CC(OC)C2)n[nH]c2c1CSCC2 66229,c1(OC2(C)CCC2)cccc(Br)c1.C1(=O)COCC(=O)NCCN1C(C)C 66230,c1(C(=O)NCC(C)NC(C2CCCC2C)=O)ccc2c(c1)B(O)OC2 66231,N1(C(C(C)Cc2ccccc2)=O)CCC(CN(C)C(c2cnc(O)n2C)=O)CC1 66232,CC1CN(C(c2cc(CNC(c3ccon3)=O)[nH]n2)=O)CCC1O 66233,C1(C(N2C(CN(C(=O)C(CC(C)C)OC)CC)CCCC2)=O)CCCCCCC1 66234,C1(C(=O)NCC2(CCNC(c3cc(OC)n[nH]3)=O)CC2)CCCC1S(C)(=O)=O 66235,N1(C(C(C)OC)=O)CC(NC(c2ccc(F)c(C(F)(F)F)c2)=O)CC2(CC2)C1 66236,C(C(F)C(=O)NCC(O)CCNC(C1(C#N)CCC1)=O)N(CC)CC 66237,C1(NC(c2cc(CC)nnc2C)=O)CC2CCC1C(NC(=O)CN1CC=CC1)C2 66238,C(=O)(C(C)(C)CC1CC1)NCC1(N(C(=O)C=CCF)C)CC1 66239,C1(C(=O)NC(C)CNC(c2cncc(Cl)c2)=O)CCC2(CC1)CC2(F)F 66240,N1(C(C(c2cccc(C)c2)O)=O)CC2CC(C1)C2NC(C1CC1C)=O 66241,c1(C(=O)NC2CC(O)(CNC(=O)CC3CCC=CCC3)C2)ncnc2ccsc12 66242,C1(C(=O)NC(CNC(=O)C=Cc2ccncc2)C2CCC2)CCC2(CCC2)O1 66243,c1(NC(c2ncccc2NC(c2ccnc(Cl)c2F)=O)=O)cc(Cl)cc(Cl)c1Cl 66244,C1(NC(=O)C=Cc2ccsc2)(CO)CCN(C(C2CCC(=O)N2)=O)C1 66245,N1(C(CC(C)CF)=O)C2CCC1CN(C(=O)Cc1cc3ccccc3o1)CC2 66246,C1(C(=O)NC2C=CC(CC(=O)N(CCCC)CC)C2)C2CC3C(C2)C13 66247,N1(C(CC2CCN(C)C2=O)=O)C2CCC1C(F)C(NC(c1ccc(Cl)cn1)=O)C2 66248,CCC(CC(=O)N1CCCC(N2CC(C)(C)C2)C1)c1ccccc1 66249,N1(C(CCOC(C)C)=O)CC(CNC(=O)CNC(=O)C(F)(F)F)CC1C 66250,c1(CC(=O)N(C)CC2N(C(c3cc(C)ns3)=O)CCC2)ccccc1C(N)=O 66251,C1(CC(=O)NCC)OCCCC1(C)C.C=CCC(C)(C)N1C(=O)c2ccoc2C1 66252,C1(CN(C)C(c2conc2CNC(=O)COCCF)=O)COC(=O)N1 66253,C1(C(C)C)CN(C(C2CCC3(CCC3)C2)=O)CCN1C(c1cncs1)=O 66254,Cc1noc(N)c1C(N1CCC1CNC(=O)Cc1ccc(F)nc1)=O 66255,C(CC(C)C(=O)N1CCC(NC(=O)CC2CC(SC)C2)C1CC)=CC 66256,N1(Cc2ccc(C)c(O)c2)CCC2(CCCC2C(=O)Nc2cncc(CO)c2)C1 66257,Cn1nc(C(=O)NCC2CCC2C(=O)NC(CC(N)=O)C2CC2)cc1F 66258,N1(CC(=O)NC2C(CNC(CCC(C)(F)F)=O)C2)C(=O)NC2(CCOCC2)C1=O 66259,N1(C(CCC(=C)C)=O)CCCC12CCN(C(=O)Cn1cc3ccccc3n1)CC2 66260,CC(C)(C)C(C#N)C(=O)NC1COCCC1NC(c1cnc(S)n1C1CC1)=O 66261,C1(CCC(=O)OC)CC(OC)N(C(=O)C(c2ccc(C(N)=O)cc2)O)C1 66262,C(=O)(C1=NOC(C)C1)NCCC1(C(N(C)Cc2nc(C)sc2)=O)CCC1 66263,n1(CC(=O)NCC2N(C(C3ON=C(C)C3)=O)CC(O)C2)cnc2sccc2c1=O 66264,N1(C(CCc2scc(C)n2)=O)CC(NC(=O)C(c2ccccc2Cl)O)C(C)(C)C1 66265,N1(C(c2c(O)ccc(CC)c2)=O)CC2CCC(C1)N2C(C12CCCCC1C2)=O 66266,N1(C(Cc2c(C)ocn2)=O)CC2(CCN(C(=O)C(c3ccc(O)cc3)(C)C)C2)C1 66267,N1(C(=O)CC(O)C2CC2)CCCC2(CCN(C(c3ccc(O)nc3Cl)=O)CC2)C1 66268,CC1COc2c(C(=O)N(CCCCN(C)C(C3C=CCCC3)=O)C)cccc21 66269,C1(C(=O)NCC(CO)NC(c2c(COC)nn[nH]2)=O)CC2C(C1)C2(F)F 66270,c1(N(C(=O)CCN(C)C)CC2N(CC)CCC2)ccccc1Br 66271,C(N=c1[nH]c(=NC)[nH]c(=NCCSc2ccccc2)[nH]1)c1cnc(CC)s1 66272,CC#CCCCC(=O)N1CCC1CC(=O)NCC1(OC)CCC1 66273,N1(C(CSC)=O)CC(C(=O)N(C)Cc2ccsc2)C(C)C1 66274,C1(OCC)CC2(C1)CC2C(=O)NCC(C)CN(C)C(c1sc(C2CC2)nc1C)=O 66275,c1(OC)ccc(CNC2CCN(Cc3ccccc3)CC2C)c([N+](=O)[O-])c1OC 66276,c1(OCCN(CCCn2cc(C3CCCC(C(=O)O)C3)nn2)C)cncc(C#N)c1 66277,c1(C(N(CCN(C(C23CC(C)C2C3)=O)CC)CC)=O)cnn(-c2nccs2)c1 66278,c1(NC(C2C3CN(C(Cc4c(C)noc4C)=O)C2C3)=O)cnc(C#N)nc1 66279,c1(C(CC)C)nc(C)cc(=NC2CC(NC(=O)CC3CC4CCC3C4)C2)[nH]1 66280,C1(NC(=O)CC2CCCC(OC(F)F)C2)CCCN(C(c2cnn3cc[nH]c23)=O)CC1 66281,N1(Cc2c(C(=O)OCC)n[nH]c2)c2cccc(O)c2CCC1C 66282,N1(C(C2(CC#C)CCOC2)=O)CC2CC(NC(c3c[nH]cc3C3CC3)=O)CC1C2 66283,Cc1[nH]nc2c1CC(C(N1CCC(CO)(NC(=O)Cn3cccn3)CC1)=O)CC2 66284,n1(CC=C)nnnc1C(CC(C)C)NC(C)CC(=O)Nc1ccccc1 66285,C12(CNC(C(C)=C3CC3)=O)CCC(C1)N(C(=O)CSCC(F)(F)F)C2 66286,c1(C(=O)NC(C(=O)N(CCNC(c2cccs2)=O)CC)C)ccccc1Cl 66287,c1(CC)ncc(Cl)c(C(N2CCCC(NC(=O)COC3CCCCCC3)C2)=O)n1 66288,C1(CC(N2CC(NC(c3cn(C)nn3)=O)CC2(C)C)=O)Cc2ccccc2C1=O 66289,CCCC(CC)CCC(=O)N1CCC(N(C)C(c2cc(N)ccc2O)=O)C1 66290,c1(C(=O)NC2C(C)N(C(c3cnc4sccn34)=O)CC2)ccc([N+](=O)[O-])s1 66291,CC1CC2CCC(C(=O)NCCC(C)NC(c3ncc(Cl)n3C)=O)CN2C1 66292,c1(OC)cc(C(=O)NC2CCC(NC(c3ccncc3C3CC3)=O)C2)ccc1F 66293,c1(C(=O)NC2CCNCC2F)cnc2c(cnn2Cc2ccccn2)c1 66294,c1(C(N2C3(CNC(CC=CC=C)=O)CCC3CC2)=O)cnc2c(c1)NCC(=O)N2 66295,c1(CC(=O)NCC2C(NC(c3cncc(C)c3Cl)=O)C2)cccc2nsnc12 66296,N1(C(C(C2CCOC2)OCC)=O)C2CCC1CC(CNC(C1CC(F)(F)C1)=O)C2 66297,CC1CN(C(C2(C#N)CCCO2)=O)CC1CC(=O)NCC(C)S(N)(=O)=O 66298,CC1CCCC(NC(=O)CCc2nnc(CSc3cccc(C(F)(F)F)c3)s2)C1 66299,N1(C(CCSCCCC)=O)CCC(CO)C(NC(=O)CC2CCCCC2(C)C)C1 66300,Cc1cnccc1C=CC(=O)NCC1(CN(C)C(c2cc(O)n(C)n2)=O)CC1 66301,Cc1cc(C(=O)NC2(C)CC(NC(c3cc(Cl)no3)=O)C2)nc(O)n1 66302,C(=O)(C1=C(C)CCC1)NC(C(N1CC(CCC#C)C1)=O)C1CC1 66303,C1(NC(CCCOC)=O)CCC(NC(C23CC(CN2C2CC2)C3)=O)CC1 66304,C12(CNC(C(C)(C)OC)=O)CCCN(C(=O)C=Cc3cccc(F)c3)C1C2 66305,C1(C(=O)NCCC)CC2CCN(CCCN3CCC(CN(C)C(C)=O)CC3)CC12 66306,C1(C#N)(C(=O)NCC2N(C(CCC(CC)OC)=O)CC2)CC2C=CC1C2 66307,C1(C(=O)NCCCCN(C)C(C23CCC(C)(CC2)C3)=O)CC12CCCOC2 66308,C1(C)(C(=O)NC(CN(C(c2ccccc2SC)=O)CC)C)CC(OC)CN1C 66309,C1(NC(=O)OC(C)(C)C)CN(Cc2cc(Br)cc(Br)c2O)CC2(CCOCC2)C1 66310,CN1CCCCN(C(c2cnc(C(C)(F)F)s2)C(=O)NCCC2(C)CC2)CC1 66311,C1(NC(c2nc(CCCCC)sc2)=O)CCCC(N(C)C(c2ccnn2C)=O)C1 66312,N1(C(c2nc(CC)sc2)=O)CCC2CCN(C(C3(C)CC3C)=O)CC12 66313,C#Cc1cccc(NC(C2CN(C(C3(CC(=O)OC)CC3)=O)CC2C)=O)c1 66314,c1(CN(CCOC)CC2CC=CCC2)ccc(Cl)s1 66315,c1(C(=O)NC2CC(F)(CNC(CCC)=O)C2)cnc(C(F)(F)F)c(F)c1 66316,C1(N(C(C2N(C)CC2)=O)C)CN(C(C2(C)CCCC2)=O)CC1(C)C 66317,c1(CN(c2nnnn2CCCF)CC)cc(F)c(F)c(OCC2(C)CCOC2)c1F 66318,CC#CCCC(=O)NC(C)(CNC(=O)CSCC1CCCO1)C(C)C 66319,C(=O)(CCCCN=[N+]=[N-])N1CCC(C(=O)NCC(C(C)C)(C)O)(CO)C1 66320,CCC(O)C(F)(F)C(=O)NCC(CCNC(C1(n2nccn2)CC1)=O)OC 66321,C1(NC(COCCSC)=O)CCCC(NC(c2cc(-c3cccs3)on2)=O)C1 66322,N(C(=NCCCN1CCCC1)N1CCN(CCc2scnc2C)CC1)CC(=C)C 66323,CCCC(C)CCCC(=O)N(CC(C)NC(C1(c2cccs2)CCCC1)=O)CC 66324,CN=c1[nH]c(=NCc2ccc(SC(C)C)cc2)[nH]c(=NCCCNC(C)=O)[nH]1 66325,C1(CNC(CC(CC)NC(c2cnc(=N)[nH]c2)=O)=O)OC(=O)CC1(C)C 66326,C1(NC(=O)NCC(C(C)C)c2ccccc2)CC2(C1)CC21CCC1 66327,C=C=CCN=c1[nH]c(=NCC2CC(S(C)(=O)=O)C2)[nH]c2c1SCC2 66328,c1(C(=O)NC2CCN(C(c3c(C)[nH]cc3)=O)C2(C)C)ccc(Br)c(F)c1F 66329,c1(C(=O)NCC2(C)C(NC(c3c(OC)csc3)=O)CCC2)cc2c(Cl)cncc2o1 66330,c1(CC)cccc2c1CN(C(c1cc3n(n1)CC(O)CO3)=O)CC2 66331,n1(C(C(=O)NC(CCC)C(=O)OCC)CSC)ccc2sccc2c1=O.C(C)(C)C 66332,CC1CC(C)(C(=O)NC(C)CN(C(=O)CCn2ccccc2=O)C)CC(C)O1 66333,c1(C(N(C2CCN(C(C(CCC)C)=O)CC2)C)=O)ccc2nc(C)n(C)c2c1 66334,C(=O)(CCCCC(=O)NC1CN(C(c2ccc(C(C)=O)c(F)c2)=O)CC1O)NC 66335,N1(C(C(C)OC)=O)CCC(F)(CNC(=O)Cc2cncc(C#N)c2)CC1 66336,CCC(C)C(O)C(=O)NCCC(C(C)C)NC(C1CCOC(CC)C1)=O 66337,C(=O)(C1=CCCOC1)NC(C(C)NC(=O)Cc1ccc(Cl)cc1)CO 66338,C1(NC(CC2(C=C)CN(C(=O)CC(=O)N(C)C)C2)=O)COC2(CCC2)C1 66339,n1(C(C)C)ccc(CC(=O)NCC(C)NC(=O)CC(C)C2CCCCC2)n1 66340,c1(C(N2CC(CN(C(CCCC)=O)C)OCC2)=O)cc([N+](=O)[O-])oc1C 66341,c1(OC)c(C(=O)NC2CC(C)N(C(=O)Cc3cccc(Br)c3)C2)ccnc1F 66342,N1(C(c2cccc(C(C)=O)c2)=O)CCN(C(=O)C(c2ccccc2)C)C(CO)C1 66343,N1(C(C2(Oc3cn(C)nc3)CC2)=O)CCCCC1NC(=O)CC(O)C1CC1 66344,C1(CNC(c2cc(CNC(CC3(N(C)C)CCC3)=O)on2)=O)CCCC12CCC2 66345,N1(C(CC(C)C)=O)CC(C(=O)NC(C)Cc2cn[nH]c2)OC(C)C1 66346,c1(OCC(=O)NC2CC(C)CN(C(=O)CSCCN(C)C)C2)cc(F)ccc1F 66347,C1(CNC(C(C)OC)=O)CCCCCN1C(c1nc(C)ncc1Br)=O 66348,CCC(C)C(O)C(C)C(=O)NC(C)C(=O)N(Cc1ccc(C)o1)OC 66349,C(=O)(C(F)(F)C(O)C(C)C)NCC1C(NC(C2CN(C(C)=O)C2)=O)CCC1 66350,C1(COC)(NC(=O)C(C)NS(C)(=O)=O)CCN(C(C2CCCCC2O)=O)CC1 66351,c1(NC(CC)CNC(C2CCCSC2)=O)ncc(C#N)cc1Cl 66352,C(=O)(CS(=O)(=O)c1ccccc1C)NCC(CNC(c1cncc(CC)c1)=O)O 66353,C1(NC(=O)CCCc2ccncc2)CCCN(C(C2CC23CCCC3)=O)CC1 66354,C1(c2n(CC=C)nnn2)(NCC2(C3CC3)CC2)CCOC(C)C1 66355,CCC(CCCC(=O)NCc1cnn2ccccc12)NC(=O)CSC 66356,CN1CC2CCN(C(=O)C=CCNC(=O)CN3CCOCC3)C2C1 66357,C(=O)(C(CC(N)=O)NC(=O)CC(C)CN(C)C)NC(COC)C(C)C 66358,C(=O)(N=c1cc(OC)n(C)[nH]1)C1(C(=O)NCCOCC#C)CCN(COCC)CC1 66359,C1(C(=O)NC(c2cn(-c3c(C)ccc(C)c3)nn2)C)CCc2nc(C)sc2C1 66360,c1(C(=O)NC2C(NC(=O)CC3C=CCCC3)CCC2)ccc2c(c1)CC(=O)NC2 66361,Cc1cc(C(N2CCC(N(C)C(c3cncc(NS(C)(=O)=O)c3)=O)C2)=O)ccn1 66362,CCCCCC(=O)N1CCC(C(=O)N(Cc2ccccc2)OC)C1 66363,CCCCCCC(F)C(=O)NCC(C)(C(C)C)NC(c1cc2ncccn2n1)=O 66364,C1(C(=O)NCCC(CC)(C)NC(=O)CC2CC2)CNC(=O)CN1C(=O)OC(C)(C)C 66365,Cc1ccc(CC(N2CCCC(N(C(=O)C(C)CO)C)CC2)=O)c(C)c1 66366,Cc1cccc2[nH]cc(C(N3CCCC(CC(=O)NCc4ccccc4)C3)=O)c12 66367,CCCC(CCC)CC(=O)NCC1CN(C)CCN1C(C12CC(F)C1C2)=O 66368,C(C(C)(C)C(=O)N1CCC(C)(CNC(C2(c3cnn(C)c3)CCCO2)=O)C1)OC 66369,c1(C(N2CCC(CNC(C3(C)CCCC3)=O)C2)=O)cnc(Cl)c(Cl)c1 66370,CC1(C)CC(=O)CCC1C(N1CCCC(C)(NC(=O)CCCCC2CC2)C1)=O 66371,N1(C(Cc2ccn(C(C)C)n2)=O)CC(NC(c2cc(C(N)=O)no2)=O)CCC1C 66372,C1(NC(=O)CC2CCC(O)C2)CN(C(=O)Cc2cccnc2O)C2(CCCC2)C1 66373,C(=O)(C(CC)C(F)(F)F)NC(CC=CC(=O)N(CC(=O)NCC)CC)(C)C 66374,Cc1ccc(C)c(OCC(=O)NC2CC2NC(=O)C(C(C)(C)C)c2cc[nH]n2)c1 66375,c1(C(=O)NC2CCN(C(c3nc(OC)c(C)s3)=O)CC2O)ccc2c(c1)COC2 66376,C1(NC(C(C)OCCOCC)=O)CC(OC)CN(C(=O)Cc2ccsn2)C1 66377,CCCCC(F)C(=O)NC1CCC(C)(CNC(c2cnoc2C)=O)C1 66378,c1(CC)nn(C)c(Cl)c1C(=O)NCCCC1(NC(c2cnc(O)c(F)c2)=O)CC1 66379,N1(C(C2C(C)(C)COC2)=O)CCOC2(CCN(C(=O)CCc3cnoc3)C2)C1 66380,C1(N(CCC(=O)NC(c2ccco2)C)C(C2CCO2)=O)C2CCC1CNC2 66381,c1(C(N2C3CN(Cc4ccc(OC)cc4OC)CC32)=O)cc(Br)cc([N+](=O)[O-])c1 66382,c1(N(C)C)cccc(CCC(=O)NCC2CCCN2C(=O)C(F)C2CCOC2)c1 66383,N1(C(c2cccc(OC)c2OC)=O)CC2C3CCC(C2C1)N(C(C)C)C3 66384,N1(C(c2ncc(F)cn2)=O)CC2(CCCN(C(c3ccnc4c3CCC4)=O)C2)C1 66385,C1(NC(NCCC(C)=O)=NCCCCC2CC2)Cc2n[nH]cc2C(C(F)(F)F)C1 66386,C(CC(C(C)C)NC(=O)Cn1cc(CO)nn1)NC(COCc1onc(C)n1)=O 66387,c1(C(=O)NCc2c(O)ncc(C)c2)coc2c1CN(C(=O)C(C)C1CC1)C2 66388,c1(C(=O)NCC2N(C(c3c(OC)ccnc3OC)=O)CC2)cnn2ccccc12 66389,C1(NC(CCOCCN(C(C2CC(C)(CC)C2)=O)C)=O)CCc2nncn2C1 66390,N1(C(Cc2c(C)occ2)=O)CC(CNC(c2ccsc2C#N)=O)CC1C 66391,C1(CNC(c2c(C(C)C)nn(C)c2)=O)CCN(C(c2cc(O)n(C)n2)=O)C1(C)C 66392,Cc1cn(C)nc1C(=O)NCC1CN(C(c2ccc(CO)o2)=O)CC1C(F)(F)F 66393,C1(NC(CC)=O)COC2(C1)CN(C(C1(C)CCCOC1)=O)C2 66394,Cc1cc(F)c2ncc(C(N3CC(CCNC(c4conc4C)=O)C3)=O)cc2c1 66395,C1(F)(CNC(CCCOCCC)=O)CCCN(C(C2CC2CN(C)C)=O)CC1 66396,C1(n2cc(C3CCN(C)C3)nn2)CON(C(=O)C2C3CCC(C3)C2c2cn[nH]c2)C1 66397,C1(NC(C(N2CCC(C)(C)C2c2ccccc2)=O)=O)CC12CCc1ccccc12 66398,c1(N(C)C)ccc(C(N2CCC(NC(C3(C)CS(=O)(=O)C3)=O)C(F)C2)=O)cc1F 66399,c1(CN2CCCC(C)(C(=O)NCC=Cc3cccs3)C2)ccc2c(c1)CNC2=O 66400,C1(CCOC)CN(C(=O)CC2CCCC(C)(C)C2)CCN1C(c1cc(F)n[nH]1)=O 66401,c1(C(N2CCC(OC)(CNC(c3ccc(C)c(F)c3)=O)C2)=O)cc(C)cc(Cl)c1 66402,C1(NC(c2cn(C)nc2Br)=O)CN(C(=O)CCc2ncc[nH]2)CC(C)(C)C1 66403,c1(C(=O)NCCCCNC(CCCC(CCC)C)=O)sc2nccc(C)c2c1C 66404,N1(C(c2ccn(CC(C)C)n2)=O)CCC2(CCN(C(C3(C)CCCS3)=O)C2)C1 66405,c1(-c2cn(CC(=O)NCc3ccc(-n4cncn4)cc3)nn2)cccnc1Cl 66406,C12(NC(C(n3c(C)ccn3)C)=O)CCCC(NC(=O)C3=COCC3)(C1)C2 66407,c1(CNC(C(C)n2cccn2)=O)ccoc1C(N1CC(N2CCC2)C1)=O 66408,N1(C(CC2CC(CC)C2)=O)CC2C(C(N3CCCC(CCCO)C3)=O)C2C1 66409,c1(C(N2C(C)(C)CC(C(N3C4CSCC3C4)=O)C2)=O)cnc2ccccn12 66410,c1(CNC(C)=O)ccc(C(=O)NC(C)CCNC(c2c(Cl)cnn2CC)=O)cc1 66411,S(=O)(=O)(c1ccc(Cl)nc1)N1CC2C(CC(=O)Nc3ccc(Cl)cn3)C(CC2)C1 66412,N1(C(C2(C#N)C(C)C2)=O)CC=C(C(=O)NCc2cocn2)C1 66413,N#Cc1ccc(C=CCOC(C23CC(CC4CC4)(CO2)C3)=O)cc1 66414,c1(CCC(N2CCN(C(C(CC)SC)=O)CC2C)=O)cccc2oc(C)nc12 66415,C1(CNC(c2n(CCOC)ncc2)=O)C(C)CCCN1C(=O)C=Cc1ccsc1 66416,N1(C(Cc2cnc(C)s2)=O)CCCC(O)(CNC(C2CC2C(F)(F)F)=O)C1 66417,CCC(C(=O)N1CC(O)(COC)C1)N(C(=O)C(C)C1(O)CCC1)C 66418,N1(C(CCNC(=O)CO)=O)CC(O)(C(F)C(=O)N(C2CC2)Cc2ncccn2)C1 66419,CCC(CC(F)F)C(=O)NC1(C(C)(C)C)CCN(c2ccc(C#N)c(C)n2)C1 66420,c1(NCc2c(OC)cc(C#N)cc2)nc2ccccc2nc1NCCC(C)OC 66421,c1(-n2cc(C3(N(C)C)CN(C(=O)CCN4CCC4)C3)nn2)c(F)cc(Cl)cc1F 66422,C(c1ccsc1)=CC(=O)NCCN(CCOC)C(c1nscc1C)=O 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66494,C12(C(=O)NCc3cc(C)ncc3)CC(CN(C(C3CCSC3)=O)C1)C2 66495,N(C(=N)N1CCC(Cc2ccccc2)C1)C(C)CC#N 66496,N1(CC(CC)OC)CCCC(CO)(NC(c2cnn(C(C)C)n2)=O)C1 66497,Cc1cccc(C)c1SCC(N1CCCC(N2CC(F)(F)C2)C1)=O 66498,C(CC(C)C(=O)N(C1CCCCC1NC(=O)Cc1ccsc1Br)C)=CC 66499,N1(C(c2cn(CCNC(c3c(CC)nccc3)=O)nn2)=O)CCCC(CC)CC1 66500,C1(CCC(=O)N(CCNC(C(CC)OC)=O)C2CC2)CC(C)(C)CO1 66501,CC1CN(C(=O)C=CCF)CCC1NC(c1nn(C)nc1Br)=O 66502,c1(SC)cc(C)ccc1C(=O)NCCN(C(c1ccn(C2CC2)n1)=O)CC1CC1 66503,Cc1cc(C(=O)NC2CSC(C)C2)nc(N(C)C)n1 66504,N1(C(c2c(CCC)nns2)=O)Cc2nccn2CC(NC(=O)C=C(Cl)Cl)C1 66505,c1(C(N(CCCNC(=O)C2=COCC2)CCO)=O)ccc2nn[nH]c2c1 66506,N1(C(CC=CCCCCC)=O)CCCC1C=CC(=O)NC(c1nnc(C)o1)C 66507,C1(CC(=O)NC2(CNC(=O)Cc3cccc(Cl)c3)CCOC2)CCCC1(F)F 66508,C1(NC(C2(COC)CN(C(c3cnc(S)nc3)=O)C2)=O)CCN(C)CC1C#N 66509,c1(C(=O)NCCC2CCN(C(CCOCC)=O)C2)scc(C)c1OC 66510,C1(NC(C(c2ccncc2)C)=O)CCC2CC1CN2C(C1CCCNS1(=O)=O)=O 66511,n1(CC(=O)NC2C(SC)CN(C(C3(C)CCCO3)=O)C2)cnc([N+](=O)[O-])c1 66512,CC1(C)CCCCC1C(=O)NCC1CC(NC(C2CCC23CCC3)=O)C1 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66531,C(C(C)(CC)C(C)O)NC(C1(CNC(=O)CC=C(Cl)Cl)CC(=C)C1)=O 66532,c1(C(=O)NC(CC(F)F)C(=O)NCC(Cl)=CCl)ccc2n[nH]cc2c1 66533,c1(CC(=O)NCC(C)CN(C(=O)C(C)(C)C2CCCC2)C)ccn(C(F)F)n1 66534,N1(C(c2c(COC)scc2)=O)CC(O)C(O)C1CNC(C1CCC2CC12)=O 66535,N1(C(C(CC)(C)O)=O)CCCCC(CNC(=O)CCc2csc(=N)[nH]2)C1 66536,N1(C(C(=O)NCCOC)=O)CCN(C(=O)CCNC2CCN(C)CC2)CC(O)C1 66537,Cn1cccc(C(=O)NC2CC(CCNC(C3CC3(C)C(F)F)=O)C2)c1=O 66538,C#Cc1cccc(CC(=O)NC(CCC=C)C(=O)N(CC2=CCCOC2)C)c1 66539,Cc1ccccc1-n1nc(CC2CC2)nc1-c1cnc(C(C)(C)C)nc1 66540,c1(NC(C2C(C(=O)Nc3ccnc(C)n3)C2)=O)ccc2c(c1)C(=O)NCC2 66541,C(=O)(C1=NOC2COCC12)NCC1(F)CCC(NC(c2c(C)oc(C)c2C)=O)C1 66542,N1(C(CCC=CCCC)=O)C(CNC(=O)C(C)SC)CC2CCCC12 66543,c1(N(CC(=O)N(C)CCNC(C2(C(C)(C)C)CCC2)=O)C)ccc(Cl)nn1 66544,C(=O)(CCC(C)(C)N(C)C)NCC1(C(=O)NC2C(C)N(C)CC2)CCCO1 66545,c1(C(N(C(CCNC(c2cc(C(C)C)[nH]n2)=O)C)C)=O)cc2cccn2c(O)n1 66546,C1(CNC(Cc2ccn(CC(C)C)n2)=O)CCN(C(=O)COCCCF)C1(C)C 66547,CCC(C)C(C)(O)CNC(=O)C(C)(CNC(c1ccc(C)n1C)=O)CC 66548,N1(C(C(CC(C)C)C)=O)CCCC2CN(C(C3(F)C(C)(C)C3(C)C)=O)CC12 66549,C(=O)(C1=C(C(F)Cl)N(c2ccccc2)C(=O)NC1c1cnc(C2CC2)[nH]1)OCC 66550,c1(C(C)C)nccc(C(=O)NC2CC(NC(=O)Cc3ccc(Br)cc3)C(O)C2)n1 66551,c1(C(=O)NC(C2CN(C(C3(C)CCCCO3)=O)C2)C)ccc(F)c(F)c1F 66552,S(=O)(=O)(c1cccnc1N1CCc2oc(C)nc2C1)NC(CCC)CC 66553,c1(NCc2cccc(C(N)=O)c2)ncccc1S(=O)(=O)N1CCC2(CCCC2)C1 66554,CC(F)(F)CN=c1[nH]c(=NCC2(CCO)CCOC2)[nH]c2c1COCC2 66555,c1(SC)cccc(C(N2CCC(NC(=O)CN3CCC(O)CC3)C2)=O)n1 66556,c1(CC(N2C(CNC(C3CCCOC3)=O)C=CC2)=O)c[nH]c2ccc(Cl)cc12 66557,N1(C(C)=O)CCCC2CCN(C(=O)C=CSCc3ccco3)CC12 66558,c1(C(=O)NCCC(C)N(C(c2cn(CC=C)nc2)=O)C)cc2cccnc2s1 66559,c1(C(C)C)ccc(C(=O)N(CC(C)NC(c2c(Br)nnn2C)=O)C)c(O)n1 66560,N1(C(C(CCSC)O)=O)CC(C(N2CCCC2C(=O)N(C)C)=O)OC(C)C1 66561,C1(C(N2CCC(n3cc(CN(CC)CC)nn3)C2)=O)CCC(N=[N+]=[N-])C1 66562,N1(c2ccc(SC)s2)CCN(C(=NCC(=O)NC(C)C)NCCCC(F)F)CC1 66563,c1(C(=O)NCC(CNC(C(c2cccs2)SC)=O)C)cn(C)c(=O)n(C)c1=O 66564,C(=O)(C(CCOCCO)NC(=O)Cc1cccc(O)c1)NC(CC(=O)NC)C 66565,c1(NC(C)CCCOc2cccnc2)ccc(CO)cc1.C12CCCN1C2=O 66566,CC1=CCSC1C(=O)NCC1CCCCO1.C12CCC1C(=O)NC2 66567,c1(C(N2C3C(NC(C4(C#C)CCC4)=O)CC(C3)C2)=O)cc(F)c(OC)c(F)c1N 66568,C1(C(=O)NCC(CCNC(C(CC)COC)=O)OC)OC(C)(C)OC1(C)C 66569,N1(C(CC(C)N(C)C)=O)CCC(C)(C(=O)NCCCC(N)=O)CC1 66570,N1(C(COCC)=O)CCC(CN(C(=O)C(C2CCOC2)OCC)C)CC1 66571,N1(C(C2(CC#C)CCOCC2)=O)C2CCC1CC(NC(=O)Cc1csc(S)n1)C2 66572,c1(C(=O)NC2CCC(C(N3CCCC(F)(CO)C3)=O)C2)cc2ccccc2o1 66573,C1(C2CCCO2)(C(N2CC(C(C)NC(COCC=C)=O)C2)=O)CCCO1 66574,Cc1ccc(F)cc1CC(N1CC2(C)CC1C2NC(C1CCC1)=O)=O 66575,N1(C(c2c(C(=O)OC)c(C)[nH]n2)=O)CCC(NC(c2cnc[nH]2)=O)C(F)C1 66576,c1(C(=O)NCCC2(CNC(C3(C#N)CCCO3)=O)CC2)coc2c1C(=O)NCC2 66577,c1(C(N2CCC(C(C)NC(CCC(=C)Cl)=O)C2)=O)cncc(Cl)c1C 66578,c1(N2CCC(CCN(C)C)C2)nc(N(C)CC2(OC)CCC2)nc2c1ncn2C 66579,CC(CCC(=O)NC(c1ccccc1)C)NC(C1CNC(=O)O1)=O 66580,C(c1cccnc1)=CC(=O)N(CC(C)NC(c1c(C)c[nH]n1)=O)CC.C(C)C 66581,c1(N)cncc(C(c2cn(CC(C(=O)N3CCCC3C(=O)O)F)nn2)=O)c1 66582,C=C1CC2CCCC(C1)N2C(Cc1ccccc1)CCc1ccccc1 66583,N1(C(CCCc2onc(C)n2)=O)CC(NC(c2c(Cl)c(C)nn2C)=O)CC(C)C1 66584,c1(CN2CC(C(=O)Nc3ccc(N(C)C)cn3)C(O)CC2)ccc(C#N)c(F)c1 66585,C1(NC(C(c2cncnc2)C)=O)CN(C(=O)C(N)=O)Cc2nccn2C1 66586,C12(C(N3CCC(NC(c4cn(CC=C)nn4)=O)C3)=O)CCOC(C)(C1)C2 66587,Cc1ccc(OCC(=O)NCC2CC(CNC(c3cncc(Cl)c3)=O)CO2)cc1 66588,C(=O)(CCCCc1ccc(F)cc1)NCC(C)(CO)NC(=O)CCc1ccco1 66589,c1(CC)cc(C(=O)NCc2cn(CCNC(=O)CCc3cn[nH]c3)nn2)ncn1 66590,C=CC1OCCC1C(N1CCC(CN(C)C(c2ocnc2C)=O)C1)=O 66591,CC1(C)CCCCC1=CC(=O)NC1CC2(C1)CC(CNC(=O)C(F)(F)CO)C2 66592,C1(C(=O)NC2(CCOC)CCN(C(=O)Cc3cnsc3)C2)CC2C=CCC(C1)C2 66593,c1(C(C)NC(C(COCC)NC(=O)C(C)C2CCCC2)=O)cccc(C)n1 66594,C(=O)(C(C(C)(C)C)n1cc(C2CCCCCC2)nn1)NCC(C)CC1CCC1 66595,C1(C(N2C(C(=O)OC)C3CC3C2)=O)CC12CCN(C(C1(C(=O)N(C)C)CC1)=O)CC2 66596,CC(C)C1=NOC(C)(C(N2CC=CC(NC(=O)Cc3cccc(F)c3)C2)=O)C1 66597,N1(C(CC(C)SC)=O)CCC(O)C(NC(C2SC3C=CC2CC3)=O)C1 66598,N1(C(C(CC2CCC2)OC)=O)CCS(=N)(=O)C(C)C1 66599,C1(O)(C(C)NC(=O)C=Cc2cc[nH]n2)CCN(C(c2nncs2)=O)C1 66600,C1(NC(C2OCCC(C)C2)=O)COCCN(C(C2CCCSC2)=O)C1 66601,Cc1cc(CC(=O)N(C2CCN(C(C3CC(C)(C)C3)=O)CC2C)C)cc(F)c1 66602,C1(CC(C)NC(c2n(C(CC)C)ncc2)=O)CCN(C(C2CCC(C)O2)=O)CC1 66603,C(=O)(C(C(C)(C)C)NC(C1CC12CCN(C(c1nonc1N)=O)C2)=O)NC 66604,c1(C(N2CCC(=CC(CC)C)CC2)C(=O)NCCCSC)ccc(F)nc1C 66605,C#CCCCC(=O)NCC1(CNC(c2ccc(C(C)=O)o2)=O)CC12CCC2 66606,C(=O)(C(C(C)(C)C)n1ccnn1)NCCN(C(CN(CCC)C)=O)CCCN(C)C 66607,C1(CCC=C)(C(=O)NCc2sccc2C)CN(C(=O)CCn2ccnn2)C1 66608,CCC(CC(=O)N(C1CCCN(C(=O)CCC(F)F)C1)CC)SC 66609,C1(C(=O)OCC)C2CC(NCCOC(F)F)CC12.c1(N)ccccc1OC 66610,C1(NC(c2cc(C)ns2)c2nnnn2C2(C)CC2)CCc2ccccc2C1 66611,CC(C)C(C(=O)NCC1CN(C(=O)CN2CCCCC2=O)CC1O)N1CCCC1 66612,C1(NC(C2CCCN(C(C3(OC)CCCOC3)=O)C2)=O)CC=C(C(C)C)CC1 66613,c1(CC(=O)NC(C)(C)CNC(c2cccc(CF)c2)=O)ccc2c(c1)COCC2 66614,c1(C2(C(=O)NCCCNC(=O)C(O)CN3CCCC3)CCC2)c(F)cccc1F 66615,C1(CC)CCC(C(=O)NCC2(C(=O)NCc3nc(C)cs3)CCCC2)O1 66616,c1(OC)cc(Cl)ccc1C(N1CCCCC1CNC(C1(CO)CC(F)(F)C1)=O)=O 66617,N1(C(C2C=C(C)CS2)=O)CCCCC(N(C(=O)CSc2nccn2C)C)C1 66618,c1(C(=O)NCC(CNC(=O)CN2CCOCC2=O)O)cccc(F)c1O 66619,Cc1sc2ncc(C(=O)NCC(=C3CN(C(=O)C(C)(C)C)C3)F)n2c1C 66620,C=C(C)C1OCCC1C(N1CCCC(C)(NC(c2cc(C)ccc2C)=O)C1)=O 66621,c1(C(N2CC(=C(CNC(Cn3c(C)ccn3)=O)F)C2)=O)ccc(F)c(O)c1F 66622,CCC1=C(C(=O)NC(CNC(c2cn(C(F)F)c(C)n2)=O)CC(F)(F)F)SCCO1 66623,c1(CC(N2C(CNC(C(CC)(C)CC)=O)CC2)=O)cn2cc(F)ccc2n1 66624,C12(CNC(c3ncc(CC)nc3)=O)CCCCC1N(C(=O)CC1(CO)CC1)CC2 66625,c1(-n2c(C3COC(=O)N3C)nc(C(C3CC3)OC)n2)ccc(Br)c(F)c1 66626,Cc1cc(C(N2CC(CNC(C3CCCC(=O)N3C)=O)C3(CC3)C2)=O)nnc1O 66627,N(C1CCc2cccnc21)C(c1ccc(CNCc2ccc(OC)cc2)cc1)=O 66628,N1(C(C(C)Cc2ccccc2)=O)CC2(CCC2NC(c2cc(Cl)no2)=O)C1 66629,C1(C(=O)NCC(CC)n2cccn2)(NC(c2cc(CO)on2)=O)CCC(C)(C)C1 66630,C1(NC(C=CC)=O)CN(C(c2ccc3n[nH]cc3c2)=O)CC(C)(C)C1 66631,c1(OC)cc(C(N2CCC3(NC(c4nccnc4C)=O)CC3C2)=O)cc(Br)c1 66632,N12CCC(O)(C1)C(C)CNC(=O)CC1CC(C1)C2=O.C(=O)(CCN)NC(C)=O.CO 66633,c1(CC)scnc1C(=O)NC1CCC1NC(=O)CNC(c1ccoc1)=O 66634,c1(C(=O)NCC(C2CCCC2)NC(C(CCC)C)=O)ccc(OC)c(OC)c1C 66635,N1(C(C=CCCC)=O)CCC(C)C(CNC(C2(COC)CCCO2)=O)C1 66636,CCCCCCC(C)(C)C(=O)NC(CNC(c1cc(C)no1)=O)CCC 66637,N1(C(C(COCC)C)=O)CCC2C(NC(=O)CCc3cc(C)on3)C2C1 66638,N1(C(C(CC)CC)=O)CCC(C2CCN(C(=O)COC)CC2)CC1 66639,N1(C(C2CC(O)C(F)C2)=O)CC2CC(C(=O)NCCCCCO)(C2)C1 66640,n1(CC(=O)NCC2N(C(C3C(CC(C)C)C3)=O)CCCC2)cccc(N)c1=O 66641,N1(C(C2(CC#C)CCOC2)=O)CC2CCC2(CNC(=O)Cc2cnn(C)c2)C1 66642,C(=O)(C1=CCCOC1)N(C1CCCC(N(C(=O)Cn2cc(Cl)cn2)C)C1)C 66643,C1(NC(C(CC(=O)OC)C)=O)CN(C(=O)C(C(C)C)C(C)C)CC12CCCC2 66644,c1(C(N(CCNC(C(C(=O)OC)F)=O)CC2CC2)=O)coc2ccc(OC)cc12 66645,c1(CC(=O)NCC2CC(NC(=O)CC3(O)CCOCC3)C2)cncnc1O 66646,CC1CN(C(C2CCCC2F)=O)CC(C)N(C(=O)Cc2cc(Cl)cs2)C1 66647,c1(C(C(=O)NCC)N(CC(=O)Nc2cccc(C)c2)C)cn2cc(Cl)ccc2n1 66648,C(=O)(CCCC(N)=O)NC1CN(C(C=CCOC)=O)C(C)C1 66649,C1(C(=O)NC2C(OC)CN(C(C3CCN(C)C3)=O)C2)CSC(c2ccccc2)=N1 66650,C1(OC)CN(C(c2n[nH]c(C)c2Cl)=O)CC1NC(=O)CCc1nc(C(C)C)no1 66651,C1(O)(CCNC(CC#N)=O)CCCN(C(c2cccc(C(F)(F)F)n2)=O)C1 66652,C(=O)(C(CCC(C)C)NC(C1CC2CCC(C1)O2)=O)NCC(C(=O)OC)OC 66653,N1(C(C(CC)n2cccn2)=O)CCC(O)(CN(C)C(C2CCC=CCC2)=O)C1 66654,N1(C(Cc2nc(C)sc2)=O)CC(NC(=O)CCC(=O)c2ccc(O)cc2)C(C)C1 66655,c1(C(N2CCOC(C3CCCOC3)C2)C(=O)NCCOC)cnc(C(=O)OC)nc1 66656,Cc1cnn(CCN(C(=O)C(CN(C)C)NC(C2CC2C(N)=O)=O)C)c1 66657,c1(C(N2CCC(NC(C=C(CCC)C)=O)(CO)CC2)=O)cccc2c1C(=O)NC2 66658,C12(C(=O)NCC(C(C)C)(C)NC(c3cscn3)=O)CCCC1CC(=O)C2 66659,CC1CC(C(=O)OC(C)(C)C)CN1C(=O)Oc1c(NC(N)=O)cccc1 66660,C#CCC(CC(=O)OC)NC(=O)C(CNC(=O)C1=C(Cl)CCC1)CCC 66661,c1(CNS(c2cc(C(=O)NC)n(C)c2)(=O)=O)c(OC)ccc2cccnc12 66662,c1(C(N(C)CC2(NC(Cc3c(C)nc(C)s3)=O)CC2)=O)ccc2oc(O)nc2n1 66663,c1(NC(c2ccc(OC)s2)=O)cn(C)c(C(=O)N(C)CC2CCCCC2)n1 66664,c1(C(=O)NC2CC(NC(C3(CC)CCOC3)=O)C2)cnc2cccnn12 66665,CC1CC(NC(=O)C(C)NS(C)(=O)=O)CN(C(=O)CC=Cc2ccc(F)cc2)C1 66666,C(=O)(C(C)(CSC)NC(c1cc(Cl)cs1)=O)NCC(COC)C 66667,CC(C(=O)N1CC(c2ocnc2CNC(c2ccon2)=O)C1)P(C)(C)=O 66668,CCC(CC(=O)N1CC(CNC(=O)CN2CC3C=CC2C3)CC1C)C1CC1 66669,c1(NC(C2C(C)C2c2nn[nH]n2)=O)ccccc1C1(C)CC1 66670,c1(C(c2n(CCOC)nnn2)NC2CCOCC2(C)C)cnn(C)c1S(C)(=O)=O 66671,C1(NC(C2C(OCC)C2)=O)CN(C(c2cccnc2C(F)(F)F)=O)CC1(C)C 66672,CCC(C)CC(=O)N1CC(C(=O)NCc2cc(C3CC3)on2)C(C(C)C)C1 66673,Cc1ccc(C(=O)NC(C)CCNC(c2nc[nH]c2C(F)(F)F)=O)c([N+](=O)[O-])c1 66674,c1(C(N2CCCC(N(C(=O)C(O)P(C)(C)=O)CC)C2)=O)ccc2oc(=N)[nH]c2c1 66675,c1(C(=O)NC2COCC2NC(=O)C(O)CC2CCOCC2)cccc(C2CC2)c1 66676,C(=O)(CS(=O)(=O)C1CC1)N1CC(N(C(c2cnn(C(C)C)c2Cl)=O)C)C(O)C1 66677,C1(N(C(C(C)OCCOC)=O)C)CCCC2CN(C(=O)CCc3cccs3)CC12 66678,C1(C(C)(C)C)C(NC(=O)CC2CCC2(C)C)CCN1C(=O)CCCn1cccn1 66679,N1(C(CC23CC(C)(OC2)C3)=O)CCCCCC(NC(c2scnc2C2CC2)=O)C1 66680,C1(N(C(=O)CC2OCCC2(C)C)CC)CCCN(C(c2cc[nH]c2)=O)CC1 66681,C(CC(CC)C(=O)NC12CC1CN(C(=O)CSc1n[nH]c(=N)s1)C2)=CC 66682,N1(C(C2(C)C(C(=O)OC)CC2)=O)CCN(C(c2cnns2)=O)C(CCO)C1 66683,Cc1cccc(C(=O)NCC(C2CCN(C(=O)C(O)C(C)C)CC2)(C)C)n1 66684,N1(C(C23C(CN(c4c(C)cncn4)C2)C3)=O)CCC(O)(CF)CC1 66685,C1(CNC(C(C)NC(N)=O)=O)CN(C(=O)CC2(C#N)CC2)CCC12CCOCC2 66686,C12(CNC(CCOCCOC)=O)CSC(C1)C2 66687,c1(C(=O)NC(CCNC(COCCC#C)=O)C)cc(Cl)cc2ccccc12 66688,C(C)(C(=O)NCC1(NC(C2CC2(C)C(F)F)=O)CSC1)OCCOC 66689,Cc1nc[nH]c1CC(O)C(=O)N(CC(C)N(C)C(c1cn(C(C)C)nn1)=O)C 66690,C1(NC(C(CCSC)O)=O)CC2CCC(C1C)N2c1ncnc2onc(C)c12 66691,c1(NC(C2(C)CCN(C(=O)CCc3ccc(O)cc3)C2)=O)ccc(Br)nc1Br 66692,N1(CCN2CCCC(C(=O)OC)C2)CC(=O)CCC1=O 66693,c1(COC)ccoc1C(=O)NCC(CNC(=O)Cn1[nH]cnc1=N)CO 66694,C1(C)(CC)CCN(C(C2CCCCC2(C)NC(=O)CN=[N+]=[N-])=O)CC1 66695,C1(C(N(CCNC(=O)COc2ccsn2)CC)=O)CC(c2ccncc2)=NO1 66696,C1(CNC(CC2CCCC(C)C2)=O)CC(C)(C)CN1C(=O)CC1C=CCC1 66697,N1(C(c2c(C)n[nH]c2)=O)CCN(CCNC(C2CCC(=O)C2)=O)CC1 66698,c1(OCC(N2Cc3nnsc3C2)=O)cc(Br)cc(F)c1F 66699,C(=O)(CC(C(F)(F)F)c1ccon1)NCCCNC(C1=NOC(C)C1)=O 66700,c1(CC)[nH]nc(C(N2CC(NC(C3(C(F)F)CCCO3)=O)C(C)C2)=O)c1[N+](=O)[O-] 66701,c1(C(=O)NCc2c(C(N3CC(C)C(F)C3)=O)c[nH]n2)ccc2c(c1)CC2 66702,CC1CCOC(C(=O)N(C(C(=O)N2CC(n3ccnn3)C2)C2CC2)C)C1 66703,C1(CNC(C2C(C)CC2)=O)CCC(F)(CNC(=O)CC2CC3(CCC3)C2)CC1 66704,C1(CNC(CC(CC)C)=O)CC2(CCN(c3nc(Cl)ncc3C(C)C)CC2)CO1 66705,c1(C2(N)CCOCC2)c[nH]c2cccc(C(N3CCC4(CCCO4)CC3)=O)c12 66706,c1(OCC)ncc(C(=O)NC2CCCC2CNC(c2ccsc2OC)=O)s1 66707,C(=O)(C(C)CCCC(C)C)N(CC(CC)NC(=O)CC1CC(=O)NC(=O)C1)C 66708,CC(C)CS(=O)(=O)N1CCSC(C(N2C(C)CCC2C)=O)C1 66709,N1(C(c2cccc(C(=O)NC)c2)=O)C2CCC1CN(C(=O)C1=CC(C)(C)C1)CC2 66710,OCCCCN=c1[nH]c(=NCC2C3CCCCC3O2)c2sccc2[nH]1 66711,C12(CNC(C3N(C)CC(F)C3)=O)CCC(CC1)N2C(=O)C=C1CCCCC1(C)C 66712,C1(NC(C(CCC)O)=O)CCCCCN(C(=O)C(=Cc2ccccc2)OC)C1 66713,Cc1ccc(C)c(C(=O)NCC2(C(=O)NCC(C)CC3CC3)CC(C)(C)C2)c1 66714,C1(CNC(CC(C(C)C)C)=O)COC(C)(C)CN1C(c1cc(O)cc(O)n1)=O 66715,C1(C(=O)NCC(=O)OCCCC)CCC(C)(C)N(C(=O)CCOC)C1 66716,Cc1ccn(CC(C)(O)C(=O)N(CC(C)NC(c2ccco2)=O)C)c(=O)c1 66717,c1(C(=O)OC)cc(C(=O)N(c2ncc(F)c(C)n2)C2CCNCC2)cc(F)c1 66718,S(=O)(=O)(c1cc(C)c(Br)cc1C)NC(C1CC2(CC(OC)(OC)C2)C1)=O 66719,C#Cc1cnn(C)c1C(N1CCCC(C(=O)NCCC(C)CCO)CC1)=O 66720,C1(C)(CC)CC(NC(C23CC2CCN3C(c2sccc2F)=O)=O)CCO1 66721,c1(C(N(C)CC2(NC(c3cc(C4C(C)C4)on3)=O)CC2)=O)sccc1S(C)(=O)=O 66722,N1(C(=O)CSC(F)(F)F)CCN(C(C2(CCF)CC2)=O)CC(O)C1 66723,C1(NC(c2c(OC)csc2)=O)CN(C(c2cnc(C)[nH]2)=O)CC1O 66724,C1(C(N2CCC(CNC(C(C)C3CC3)=O)(CO)CC2)=O)CCc2nc[nH]c2C1 66725,C1(NC(=O)CC2CC2C(F)(F)F)CC(C(F)C(=O)NCCCCN2CCCC2)C1 66726,N1(C(C(CC)O)=O)CCCC(CNC(=O)Cc2ccc(OCC(F)(F)F)cc2)C1 66727,C1(NC(C2CN(C)C(=O)CC2)=O)CCN(C(=O)CCc2cnc[nH]2)CC12CCC2 66728,C1(NC(c2ccnc(Cl)c2)=O)CN(Cc2cccnc2O)CC1(F)F 66729,c1(OC)ccc(CN)cc1-c1ccc(C(=O)NCC2(N(C)C)CC2)o1 66730,CCCCC(CC(=O)NCC1CCC2(CC2)C1)NC(=O)C1=CCCCO1 66731,c1(C(=O)NC2CCN(Cc3cncc(Cl)c3)CC2F)ccc2ncsc2c1 66732,N1(C(COC(CC)C)=O)CCC(F)(CNC(C2CCC(C(F)(F)F)CC2)=O)C1 66733,Cc1cc(Cl)ccc1CC(=O)NCCC1COCCN1C(=O)Cc1cn(C)nn1 66734,C1(C(N2CCC(OCc3cn(CC(C)O)nn3)C2)=O)CN(C)NC1=O 66735,Cc1c(C(=O)NC2CCC(c3cn(CC(=O)O)nn3)CC2)cccc1C1CC1 66736,Cn1cc(C(N2CCC(C)(CNC(c3nsnc3O)=O)C2)=O)ncc1=O 66737,N1(C(CN2CCC(C)(C)C2)=O)CC2(NC(=O)COC3(C)CCCC3)CCC1CC2 66738,C(=O)(C(=O)N=c1ccn(C2CCCCO2)[nH]1)Nc1c(NC(C)(C)C)cccc1 66739,CC1(C)CCCCC(C(=O)NC2CCCN(C(c3cncc(O)c3)=O)C2)C1 66740,C1(C(N2CCCC2c2cc(C3CC3)on2)=O)CCCC2CC12 66741,Cc1cc(C(N2CCOC(CNC(C3CCN(C)C3C)=O)C2)=O)c(C)n1C(C)C 66742,c1(NC(C)=O)cccc(CC(=O)NCC(C2CCC2)NC(=O)C(C)NC=O)c1 66743,N1(C(C2(C)CCC(C)C2)=O)CC(COC(C)(C)C)C2(CCC2)C1 66744,C1(S(C)(=O)=O)(C(=O)NC(C2CCN(C(C=CCC)=O)C2)C)CCOCC1 66745,Cc1cnc(O)c(CNC(C2COCCN(C(C3(C#N)CC(F)(F)C3)=O)C2)=O)c1 66746,c1(NC2CCCN(C(C3CC4(C3)CC4(F)F)=O)C2)ncc([N+](=O)[O-])cc1Br 66747,C1(NC(c2ccc(C)s2)=O)C=CCN(C(=O)COc2cccc(O)c2)C1 66748,N1(CCC)CC(C(=O)N(CCCCNC(c2ccc(C(=O)OC)[nH]2)=O)C)CC1=O 66749,c1(OC)ccc(NC(=O)C(c2ccsc2Cl)N2CCCC2c2ccc(F)cc2)cc1 66750,N1(C(C(CC)OCC)=O)CC2CCC1C(CNC(c1cc(C3CC3)[nH]n1)=O)C2 66751,CCC(CC)CC(=O)N1CCN(C(c2csc(-c3ccccc3)n2)=O)C2CC12 66752,c1(C(N2CCN(C)C(CNC(=O)COCC3CCC3)C2)=O)cc2ccncc2s1 66753,N1(C(C(COC)N(C)C)=O)CC(NC(=O)CC(C)(C)C#N)CC12CCOCC2 66754,C1(S(N)(=O)=O)(N(CC(c2ccccc2F)NC(C)=O)C(=O)Cc2ccoc2)CC1 66755,C1(C(N(C(C(CCSC)N(C)C=O)=O)CC(C)C)=O)CCn2ncnc2C1 66756,C1(NC(CN2C(C)CC2)=O)CCC(NC(c2ccnc(OC(F)F)c2)=O)CC1 66757,c1(N2CC3CN(CC)CC3C2)nc2c(c(=NC3C=C(C)CCC3)[nH]1)COC2 66758,c1(SCC)ccc(Cl)cc1C(N1CC2C(CNC(C3CC3C(=O)OC)=O)C2C1)=O 66759,n1(CC(=O)NCC(CCNC(C2(CC)CC(C)(C)C2)=O)O)nnc2c1CCCC2 66760,N1(C(c2c(C)ccc(C(F)(F)F)c2)C(=O)NC2CC2)CCCNC(=O)C(F)(F)C1 66761,c1(C(N2CCN(C(C(CC)C)=O)CC2COC)=O)cnc2ncnc(O)c2c1 66762,c1(C(=O)NCC2CC(CNC(c3n(C)nnc3)=O)OC2)ccc2nc(S)[nH]c2c1 66763,Cc1cc(N)cnc1C(=O)NCCNC(=O)CCC1CC(C)(C)CO1 66764,CC1SCCCC1C(=O)NCC1(NC(c2cnc(O)s2)=O)CC1 66765,C=CCC(C)(C)C(=O)NCC1CCC2CC2C1.c12cn(nn1)CC(=O)NC21CCC1 66766,c1(CC)c[nH]cc1C(N1CCC(Cc2cn(C3CCC3O)nn2)C1)=O 66767,C1(NC(C2(CNCC)CC2)=O)CN(C(=O)C(CC)OCC)CC(C)(C)C1 66768,c1(OC(C)C)cc(-c2cccc(NC(c3cnn(C(C)(C)C)c3)=O)n2)ccn1 66769,CCCC(C(=O)OC)C(=O)NC(C)CN(C)C(c1sc(C)c(C)c1C)=O 66770,N1(C(C(CNC(C(COC)OC)=O)C(C)C)=O)CCC(N(C)OC)CC1 66771,N1(C(C(COCC)(C)C)=O)CC(CNC(C23CC(C)(CO2)C3)=O)CC(C)(C)C1 66772,C1(O)(C(C)C)CCCN(C(C2CCCCN2C(C2(F)CCCCC2)=O)=O)C1 66773,CC1(C)C(NC(=O)Cn2cnnc2)CC1C(=O)NCC(Cl)C(C)(F)F 66774,Cc1cc(C(=O)NC(C)CCC(=O)NCCOC(C)C)c(C)s1 66775,C(C(C)C)(C(O)C(=O)NC1CCCC(C(N2CCC(O)C2(C)C)=O)C1)OC 66776,c1(OC)cccc(Br)c1CNC(=O)OCC1CC1C 66777,C1(NC(C(C)NC(=O)NC)=O)CN(C(=O)C(F)OC(F)(F)F)CC2(CCC2)C1 66778,N1(CC(=O)NC(C=CC(=O)NC(c2ccnc(O)c2)C)(C)C)C(=O)CNC1=O 66779,C1(NC(CCCc2n(C)cnn2)=O)CCN(C(C2CC3(CCC3)C2)=O)CC1F 66780,c1(C(N2CC(CNC(CCCCCOC)=O)C(F)(F)C2)=O)c[nH]c2ccncc12 66781,C1(NC(c2ccc(C=C)cc2)=O)CCN(c2ncc(C(F)(F)F)cc2Cl)C12CCC2 66782,N1(C(c2n(C)c(C#N)cc2)=O)CCC2(CC(NC(=O)C(C)(C)c3cnsc3)C2)C1 66783,N1(C(C(C)(C)C2CCCN2C(=O)C(Cl)Cl)=O)CCCC(CCO)CC1 66784,c1(C(N2CC(CCNC(CC3(OCC)CCC3)=O)(OC)C2)=O)ccc(C)cc1 66785,c1(-n2cc(C(C)NC(C3CCCC3O)=O)nn2)ccc(I)c(Cl)c1 66786,C(C(C)(C)C(=O)NCC1CN(C(C2CCC(C)CC2)C)CCO1)OC(C)C 66787,N1(C(C(C=CC)O)=O)CCN(C(C2(CC(C)=O)CCCC2)=O)CC1CCOC 66788,c1(N2C(CCNC(=O)CC34CNC(=O)C(C3)C4)CCCC2)nc2ccccc2o1 66789,CCC(CC(=O)NC(c1ccc(CNC(C2CSCCS2)=O)cc1)C)C(C)(C)C 66790,c1(C(=O)NC2(CC)CN(C(c3ncn(CC)c3)=O)C2)ccc2cccnc2n1 66791,c1(CC(c2n(CCC)nnn2)NC23CC(F)(C2)C3)ccc(OC)c(C)c1 66792,CON=Cc1ccc(C(N2CCC3CN(C(=O)Cc4cc[nH]c4)C3C2)=O)cc1 66793,C(=O)(N=c1[nH]c(Cl)ncc1O)C1CC1C(=O)Nc1c(C)cc(F)c(C#N)c1 66794,N#Cc1ccc(CCC(=O)NC2(C(F)(F)F)CCCNC2)cc1 66795,c12ccc(cc1)NC(=O)c1scc(c1)CNC2=O.N1(CCO)CC=CC1 66796,Cc1cc(C)c(CNC(=O)C(c2ccoc2)N2CCC2C2CCOCC2)c(C)c1 66797,c1(C(=O)NCC(CO)NC(c2[nH]cc(OC)c(=O)c2)=O)ccc(C)c(Cl)c1F 66798,c1(C(N(CCNC(c2cnn(CCC)c2C)=O)C)=O)cnc2ccc(Br)cn12 66799,CC(C)CC(C(=O)NCCOCCCN(C(=O)C(O)C(C)C)C)N(C)C 66800,C1(NC(CC2(OC)CCC2)=O)CC(C)N(C(c2cc(N)ccn2)=O)C1 66801,N1(C(c2cc(OC)cc(C)n2)=O)CCC(C)N(C(C2CCCC(CF)C2)=O)CC1 66802,C12(CCNC(C(C)OC)=O)CCC(C1)N(C(=O)CCC(=O)c1ccc(C)cc1)C2 66803,C(C(C(=O)N1CCCC1C(C(=O)NC(C)(C)C)(C)Sc1cn[nH]c1)OC)OC 66804,C(=O)(C1=CCCSC1)NCCN(C(=O)C(C(=O)OC)OC)CC 66805,c1(N(CCNC(c2ccsc2C(F)F)=O)CCl)nccc(Cn2cc(Cl)cn2)n1 66806,Cc1nc(C2CCC2)oc1C(=O)NC(C)(C)CNC(C1(C#N)CC1C)=O 66807,CC1(C)C(NC(=O)C(C)(C2CCC2)NC(=O)COC2CCCOC2)C1(C)C 66808,N1(C(C2CCCC2C)C(=O)NC2CC(C3(C)CC3)C2)CCCC(C2(C)CC2)C1 66809,C1(O)(C(N2CCCC(CNC(=O)CCc3ccsc3)C2)=O)CN2CCC1CC2 66810,CCC(C)CC(=O)C(=O)N(CC(C)NC(=O)Cc1cccnc1O)C 66811,Cc1nnc(=NCCCN(C(=O)C(c2ccc(F)cc2)(C)C)C(C)C)[nH]c1C 66812,c1(COC)cc(CSc2ccccc2OCC2CCOC2)ccc1F 66813,N1(C(C(C)=C(C)C)=O)CCC(F)(F)C(CNC(c2cnoc2-c2ccco2)=O)C1 66814,CCC(C(C)(C)O)NC(=O)C(C)CNC(c1ncncc1N)=O 66815,C1(C(N2CC(F)(CC)C2)=O)CN(C(=O)CN(C2CCC2)C)CC1C1CC1 66816,n1(CC)nc(C(=O)NC2(C(=O)NCc3nccn3C(C)C)CCCC2C)cc1C 66817,N1(C(c2c(C)ncnc2C)=O)CC2(CC(NC(=O)CC3CC3)c3nccn32)C1 66818,N(C(=NCCF)N1CCC2(O)CCOCC2C1)CC1(C)CCCCC1 66819,CC1CCCCN1C(=O)CNC(=O)NCCc1cn(C)nn1 66820,c1(C(=O)OCC)ccc(CNC2CN(C(c3cnn(C)c3C)=O)C2)cc1 66821,c1(C(N2CCCC(NCC(n3cc(Cl)cn3)C)C2)=O)c(Cl)cccc1[N+](=O)[O-] 66822,C1(NC(c2nc(CC)oc2)=O)CCC2CCN(C(c3cnoc3C(C)C)=O)C1C2 66823,CC1CCC(NC(=O)C=Cc2ccc(C(N)=O)cc2)CN1C(c1nnn(C)n1)=O 66824,c1(C(N2C(C)CC(NC(c3cnc(O)o3)=O)C2)=O)cc(Br)c(C#N)s1 66825,C1(CNC(c2cc(-n3cnnn3)cc(Br)c2)=O)CC2C(O)CC2O1 66826,CC12CCCC1N(C(=O)CC1CCC1)CCN(C(=O)Cc1cnc[nH]1)C2 66827,Cc1cc(C(=O)NC2CCN(C(C3CS(=O)(=O)C3)=O)CC2C)nc2[nH]nc(O)c12 66828,C1(C)(C(=O)NCC2C(C(=O)NCC(C3CCCCC3)C)CC2)CC(F)C1 66829,C#Cc1cccc(CC(=O)OC)c1.C12(CC(c3cn(CCOC)nn3)C1)C(=O)N2 66830,C1(NC(C2C(C(C)=O)C2(C)C)=O)COC2(CCN(C(C3(C)COCCO3)=O)C2)C1 66831,c1(C(=O)NC(C)CC(C)NC(c2ncc(Cl)s2)=O)ccc(-n2ccnc2)cc1 66832,Cc1c(C(=O)NC2CC(NC(C3CCCC34CC4)=O)C2)oc2ccc(Br)cc12 66833,N1(C(c2c(C)[nH]cc2-c2ccccc2)=O)CCCC(NC(c2csnn2)=O)C1C 66834,c1(C(=O)NC2CC(F)(CNC(C3(F)CC=CC3)=O)C2)cc2cccn2c(O)n1 66835,N1(CC(=O)OC)CC(CO)OC2(CCC2)C1.c12ccc(cc1)-c1n[nH]cc1N2 66836,c1(C(=O)NCC2C(C)CN(C(C3CCOC3)=O)C2)nc2ccccc2cc1Cl 66837,C1(OCCNC(CCNC(CCC)=O)=O)CCN(C(=O)C#CC2CC2)CC1 66838,c1(CNC(C2(C)CCN2C(c2cc(Br)co2)=O)=O)cccc(F)c1Br 66839,c1(CC(=O)NCC(CNC(C2(C)CC=CCC2)=O)OC)ccccc1F 66840,c1(CC)nc(=N)[nH]cc1C(=O)NC1CCN(C(=O)C(F)C(C)(F)F)C1 66841,CC(CC(F)F)C(=O)NC1CC2CC1N(C(=O)CC(C)(C)C1CC1)C2 66842,Cc1cc(C(N2Cc3ccccc3C2)=O)c2c(c1)CCCN2 66843,C1(NC(C2C(C)(CC)C2)=O)(COC)CCN(C(=O)C=Cc2ccc(C)nc2)CC1 66844,C(=O)(CCCC(C)NC(=O)CC1CCC(=O)C1)Nc1cc(C)sc1C 66845,C1(C(=O)NCCCCNC(C2SCCS2)=O)C2(CCC2)C12CCC2 66846,N1(C(CC(C(C)C)C)=O)CC2(CNC(c3ccc4c(c3)OCO4)=O)CCC1CC2 66847,c1(C(=O)NCC2CC(OC)CN2C(C2CC(SC)C2)=O)ccc2nc(C)nn2c1 66848,CC(O)CCCCCC(=O)NCC(C1(O)CN(C(C2CC2C)=O)C1)(C)C 66849,c1(C(N2CC(N(C(Cc3cnc(C)o3)=O)C)C2)=O)cc2nn[nH]c2cc1F 66850,N1(C(C=CC)=O)CCC(CN2CCN(C(c3ccc(OC)nn3)=O)CC2)CC1 66851,C1(NC(c2cc(C(F)(F)F)on2)=O)CC2CCC(C1)N2C(c1cccc[n+]1[O-])=O 66852,Cc1cc(C(N2CCC2C(=O)NCc2cc(Cl)ccc2O)=O)cc(O)n1 66853,C1(OC)CC(C(N2CCC(NC(c3c(C4CC4)cnn3C)=O)CC2)=O)C12CCC2 66854,C1(NC(C=Cc2n(CC)ncc2)=O)C(C)CCN(C(c2n[nH]c(=N)[nH]2)=O)C1C 66855,C1(OC)(CNC(c2cc(C(C)(C)O)ccn2)=O)CCN(C(C2(C)C=CCC2)=O)C1 66856,N1(C(c2c(-n3cc(CC(=O)O)nn3)cccc2)=O)CC2CC3CCCN3C2C1 66857,C(=O)(C1=CN=C2N=CNN2C1)NCC1N(C(C2N=C(C)SC2)=O)CCCC1C 66858,N1(C(CCCC(C)NC(C2N(CC)CCCC2)=O)=O)CCC2CN(C)CC2C1 66859,c1(OC)cccc(C)c1C(=O)NCC1CN(C(=O)C(O)C(C)(C)C)CCO1 66860,Cc1ncc(C=CC(=O)NCC2CCCN2C(c2c(C)ccnc2O)=O)c(O)n1 66861,CC1(C)C(NC(=O)C2CC2)CC1CNC(N1CCC(Oc2ccccc2)CC1)=O 66862,N1(C(=O)NCC(CCSC)OC)CCCCC(OC(C)C)C1 66863,c1(CNC(=NCC2(SC)CCOCC2)NC2CC2C)ccc2c(c1)NCCO2 66864,C(=O)(CC(C(F)(F)F)OC)NC(CCNC(C1CN(CC)C(=O)CC1)=O)(C)C 66865,Cc1cc(NC2CC(NC(c3ccc(O)nc3)=O)C23CCC3)c([N+](=O)[O-])c(C)n1 66866,C(=O)(CC(O)CC1CC1)NC(CNC(C=CCC)=O)(C)Cn1cccn1 66867,C12(NC(=O)NC(CO)CCSCc3ccccc3)CCCC1CCC2 66868,Cc1noc(C)c1CC(N1CSCC1C(=O)NC1CC(C(C)(C)O)C1)=O 66869,CC1(C)CCC(C(=O)NCC2(O)CCN(C(=O)C(C)(C)c3cc[nH]n3)C2)CO1 66870,c1(C(N(C)CC2COCCN2C(=O)CCC2CC2)=O)cc([N+](=O)[O-])ccc1Br 66871,CC(C)(C)C(=O)C(=O)N1CCC(C)(NC(=O)C(CCc2ccccc2)C2CC2)C1 66872,C1(NC(C(C)(C)C)=O)CN(N2CCC(ON3CCCCC3)C2)C1 66873,c1(C(N2CC3C(NC(c4cc(C)c(N)cc4)=O)C3C2)=O)ccc2cccnc2n1 66874,Cc1nc2cccc(C(N3C(CNC(C4(O)COC4)=O)CC4COCC34)=O)c2[nH]1 66875,C1(C(=O)NC(CC2CC2)C(=O)NC2C3COCC23)CC2(CCC2)CO1 66876,N1(C(C(C=C)(C)O)=O)CC2(C1)OC1(C)CC2(NC(C2CCN3CCCC3C2)=O)C1 66877,N1(C(c2cnc(C)s2)=O)CC2CC(NC(C3CCCC(F)C3)=O)CC1C2 66878,CC1(C)CC(C(=O)NC2(CC3CC3)CC2)=NO1.C12(CC1)C(=O)N2 66879,N1(C(=O)NCCc2nn(C)c(=O)o2)CCCC(C)(C(N2CCCC2CCO)=O)C1 66880,C(=O)(CC(C(C)(C)C)NC(c1cnncc1C)=O)NC(c1ccccc1)CC 66881,C1(CC(=O)NC(C)C(C)NC(C2(N3CCOCC3)CC2)=O)(OC)CCCC1 66882,C1(C(=O)NC(C)CCNC(=O)C(O)C2CCC2)C(c2ccncc2)C1(C)C 66883,c1(NC(C2CCN2C(=O)C2=CS(=O)CCC2)=O)ccc2scnc2c1 66884,c1(NC(C2CCN2C(c2cc(Cl)cc(Cl)c2)=O)=O)ncc(F)cc1Br 66885,C12(C(=O)NC(CCNC(C3CN(C(=O)NC)C3)=O)C)CCCCN1CCC2 66886,C1(NC(c2c(CC)scc2)=O)CCN(C(c2ccccn2)=O)C(C)C1 66887,c1(C(NNC(NCN(C(C)(CC(=O)O)C(C)C)CC)=S)=O)cc(Cl)c(Br)cc1F 66888,c1(C(=O)NC2CCN(C(C3=NNC(=O)C3)=O)CC2F)ccc(F)c2ccsc12 66889,S(=O)(=O)(c1ccc(C2OCCO2)cc1)NCC1(NC(=O)OC(C)(C)C)CC1 66890,C12(C(N3CCN(C(COC(CC)(C)C)=O)C(CF)C3)=O)CCCC(=O)N1CCC2 66891,C(=O)(C(C(C)Cc1ccc(CC#N)cc1)N1CCCC(C(F)F)C1)NCCOC 66892,CCCCCS(=O)(=O)CC(=O)N1CCCC(O)(Cn2cc(CO)nn2)CC1 66893,c1(C(N(CCNC(C2C(F)(F)C23CC3)=O)CC)=O)cc(F)ccc1C(F)(F)F 66894,N1(C(C2CC(OC)(OC)C2)=O)CC2CC(NC(c3cncc(C4CC4)c3)=O)C1C2 66895,C(=O)(CC(F)(F)C(F)F)NC(c1cccc(Cl)c1)CNC(=O)CCc1cn[nH]c1 66896,C=C(C)C(C)(C)C(=O)N1CCN(C(c2c[nH]cc(Br)c2=O)=O)CC1 66897,CC1(C(=O)NCC(C)(CO)NC(c2ccc(F)cc2)=O)CC2CCC(C1)S2 66898,c1(NCCc2c(F)cncc2F)ccnc2c(Cl)cnn12 66899,CC(C)(CNC(c1cc([N+](=O)[O-])c[nH]1)=O)CC(=O)NCCCOCC(F)F 66900,C1(CNC(C(C)NC(C)=O)=O)CC2(CCC2)CN1C(=O)C=Cc1cocn1 66901,c1(NC(=O)Nc2ccc(NCc3c(C)cccc3)cn2)cc(F)cc(C)c1O 66902,C12(NC(C(C)OCC#C)=O)CCC(C1)N(C(=O)CCCC(=O)NC)C2 66903,Cc1ccc2c(C(=O)NCC3CCN(C(=O)C#CC4(C)COC4)C3)cnn2c1C 66904,C1(OC)CCC(CC(=O)NC(C)C(C)(C)NC(C2CC(=C3CCC3)C2)=O)CC1 66905,CC1CC(C(=O)N2CCC(O)(CNC(C3(F)CCCC=C3F)=O)CC2)=NO1 66906,c1(CCC(=O)NCCC2CCCN(C(C(CC)F)=O)C2)nc2cnccc2[nH]1 66907,c1(OC)ccc(CN2CCOC(CC(=O)Nc3nccnc3Br)C2)cc1[N+](=O)[O-] 66908,C1(NC(C2(C(=O)OCC)CC2)=O)CCN(C(c2ccc(N(C)C)nc2)=O)C1C 66909,N1(C(c2ccc(CC)cc2)=O)CC(NC(c2nc(C)nn2C)=O)C(C)(C)C1 66910,c1(C(N(CC(O)CNC(C2CC(Cl)(Cl)C2)=O)C)=O)cc2ccccc2c(O)n1 66911,c1(CC)cc(Cc2nc(-c3ccn(C)n3)nn2C2C(C)CCCC2C)ccc1Cl 66912,c1(NC(C(C2CC=CCC2)NC(CN(C)C2CC2)=O)=O)ccc(N=[N+]=[N-])cc1 66913,c1(CN(CCC)C(C2CCN(C(C3(c4cccs4)CC3)=O)C2)=O)ccc(Br)cc1 66914,Cn1ncc(Cl)c1CC(=O)NC12CC1CN(C(C1CC1CF)=O)C2 66915,C(C)(CC(C)(C)O)NC(C(C)N(C(=O)C(c1ccnn1C)C)CCC)=O 66916,N1(C(CSCCC)=O)CCCC(CCC(=O)N)C1.N1(CCO)CCC(C)CC1 66917,N1(C(CNC(C(CC)CC)=O)=O)CC2CCCCN2CC1CNC(=O)C=CCO 66918,C(C(O)CC(=O)N(C1CC1C)C)NC(c1c(C)ocn1)=O 66919,c1(C(N2CCC(OCCNC(C(C)SC)=O)C2)=O)ccc(-c2ccco2)nc1C 66920,CC(C)C(C(=O)N(CCCCN(C(=O)CNS(C)(=O)=O)C)C)NC(N)=O 66921,C(CC(C)C(=O)NCCCC1CCCN1C(=O)C(=O)NCC(F)F)=CC 66922,N1(C(C(C(C)(C)O)NC(C=C(CCC)C)=O)=O)CCC2(CCSC2)C1 66923,C1(CNC(Cc2nnc(C)o2)=O)CCCC2CN(C(=O)CN(C)C(C)C)CC12 66924,Cn1cc(CCNC(c2c[nH]nc2CNC(C2C=CCS2)=O)=O)cn1 66925,c1(OC)ccccc1CCC(=O)NC(C1CCCCN1C(=O)C1CC1)C 66926,C1(C)(C(N2CC3C(CNC(c4c(OC)noc4C)=O)C3C2)=O)CCC(C)CC1 66927,c1(OC)cc(C(N2CCC(NC(c3ccc(N)cc3Cl)=O)C2)=O)cc([N+](=O)[O-])c1 66928,Cc1cccc(O)c1C(N1CCCC(C)(NC(=O)CCC(F)F)C1)=O 66929,CC1CN(C(C2(c3ccno3)CC2)=O)CC(C)N(C(c2cc(O)nc(O)n2)=O)C1 66930,C1(C(=O)NCCOC2CCOC2)CCOCC1NC1CC2(CSC2)C1 66931,c1(C(N2C(C(=O)NCCCOC)C3C(C2)C3(C)C)=O)cccc([N+](=O)[O-])c1C 66932,CC1CN(C(C2CC=CCC2NC(C23CCCN2CCC3)=O)=O)CCCO1 66933,N1(C(C2(C#N)CCC2)=O)CCCC(F)(C(=O)NCCCS(C)(=O)=O)C1 66934,C(=O)(C1=CCCCC1C)N1C(C(=O)NCc2nc(C)c(C)o2)CCC1C1CC1 66935,c1(CCNS(C)(=O)=O)ccccc1NC(=O)C(=O)NCCCC1CCOC1 66936,N1(C(c2c(C)nc(COC)s2)=O)CC2(CCCC2NC(C2CCCN2C=O)=O)C1 66937,Cc1cc(CC(=O)NC23CC2CN(C(=O)Cc2ncc(C)s2)C3)cc(F)c1 66938,C(=O)(CC(C(C)C)NC(=O)Cn1c(C)ccc1C)N(CC(=O)NCCC)C 66939,C1(CNC(=O)Cc2csnn2)CC2CCC1N(C(c1csc(CO)n1)=O)C2 66940,Cc1nc(-c2cnn(C3CCOCC3N(C)C)c2)n(Cc2ccc(F)cc2)n1 66941,CCCC(CC(C)C)C(=O)NC(COC(C)C)C(N1CC(CO)C1(C)C)=O 66942,Cc1cc(CC(=O)OCC(=O)Nc2nc(C(C3CCOC3)=O)cs2)ccc1[N+](=O)[O-] 66943,c1(C(c2nnnn2CCOC)NCC(=C)C)c(OC)nsc1OC 66944,CC(C)CC(O)CC(=O)NC1(Cc2ncc(F)cn2)CC1 66945,C12(OC)CCC1CN(C(C1CCN(C(=O)CCCC3CCC3)C1(C)C)=O)C2 66946,Cc1c(NCCNC(=O)C(C)C)c(=O)n(-c2ccccc2)n1C 66947,N1(C(CC2N(C(CCC(C)OC)=O)CCC2)=O)CCc2nc(C)[nH]c2C1 66948,c1(CC(=O)N(C2CCN(C(=O)Cc3cnco3)C2)CC)nocc1C 66949,c1(C(=O)NCC2C3N(C(C=CCOC)=O)C(CC3)C2)cc(Br)cc(C)c1F 66950,O=C(CCCCCO)NC1CC(F)CN(C(c2ccc(O)c(OC(F)F)c2)=O)C1 66951,N1(C(CCCC#C)=O)CCC(C2CCCN(C(=O)CCC(=O)C(C)(C)C)C2)CC1 66952,N1(C(CCC2CCC(=O)N2)=O)CCN(C(c2cccc(Cl)c2F)=O)CC(CO)C1 66953,Cc1cccn(CC(=O)NCCCCCc2ccccc2Br)c1=O 66954,CN=c1ccc(C(N2CC(O)CC2CC(=O)NCC(=O)N2CCCO2)=O)c[nH]1 66955,O=C(CS(=O)(=O)C12CC(C1)C2)NCCCNC(c1sccc1-n1cnnn1)=O 66956,c1(NC(C2CC23CCN(Cc2c(F)ccc(Cl)c2Cl)C3)=O)nccc2[nH]ccc12 66957,CCCCCC(O)C(=O)NC(C1(O)CN(C(C2CN(C(C)=O)CCO2)=O)C1)C 66958,C1(C(N(C)C)=O)CCC(C)(C(=O)N(C)CCN(C(=O)CSCCC#N)C)C1(C)C 66959,C1(CC(=O)N(C(C)CC(=O)NCC(O)CNC(N)=O)C)CCC(=O)N1C 66960,C1(C(CO)NC(C(C)CF)=O)CCN(C(C2(F)CC2(Cl)Cl)=O)CC1 66961,S(=O)(=O)(c1cccnc1)N1CC(C(=O)NCCCNC(CN(C)C)=O)C1 66962,N1(C(c2scnc2C)C(=O)NCCCCCC)CCC2(O)CCOCC2C1 66963,c1(NCC2(CCCC)CCC2)cc(NCC2(CC3CCC3)CC2)ncn1 66964,CC(CCBr)(c1nnnn1Cc1nnc(CC2CCCO2)s1)NN1CCCCC1 66965,c1(NC(C(C)NC2(CO)CCCOCC2)=O)ccc2c(c1)OCCO2 66966,N1(C(CCCCOCC)=O)C2CCC1CN(C(c1cc(C)n(C(F)F)n1)=O)CC2 66967,N1(C(c2ccc(SC)s2)=O)CC2CCN(C(=O)C(c3cccc(F)c3)O)CC2C1 66968,N1(C(=O)OCn2nc(C)c(C3CC3)c2C)CCc2cc(Br)c(F)cc2C1 66969,C1(CNC(c2nncc(OC)c2)=O)CC2(CO1)CN(C(=O)CCc1cnc[nH]1)C2 66970,N1(C(c2c(OC)nccc2)=O)CCCN(C(c2cnc(Cl)c(Br)c2)=O)C(C)C1 66971,Cc1nc(C=CC(=O)NC2COCCN(C(C3SC4C=CC3CC4)=O)C2)[nH]c1C 66972,CN1CCCCC1CC(N1CCC1(C)CC(=O)NC1(CN(C)C)CCC1)=O 66973,c1(OCC)ccc(C(=O)NC(C2(CNC(c3cc(C#N)c[nH]3)=O)CC2)C)cc1 66974,C1(CNC(CC(=O)NCC#C)=O)CCCCN(c2nnc(C(=O)OC)s2)C1 66975,C1(C(=O)NCCN(C(=O)CCCOC2CCOCC2)CCOC)CC12CCOC2 66976,C(=O)(C1CCc2c[nH]nc21)NCC(CO)NC(c1ccn(CCF)n1)=O 66977,c1(C(C)=O)ccc(CC(=O)NCC2CC2NC(=O)C(n2cnc(C#N)n2)C)cc1 66978,C1(NC(C2CCCC23CC3)=O)CCC2(CCN(C(=O)CS(=O)(=O)C3CC3)CC2)C1 66979,Cc1cc2occ(C(=O)OCc3nonc3C)c2cc1C 66980,Cc1cc(C(=O)OC2CN(C(c3nnc(C)n3C)=O)C2)c(Cl)cc1N 66981,n1(CCCC)cc(C(N2CCC(CNC(C3CC(n4cnnc4)C3)=O)C2)=O)nn1 66982,N1(C(c2c(CC)occ2)=O)CCC(C)(C(=O)N(CCC(N)=O)C)C1 66983,C(=O)(N=c1cc(-c2ccc(F)cc2)[nH][nH]1)NCC(c1cccc(Cl)c1F)(C)C 66984,c1(COC(C2CS(=O)(=O)CC(=O)N2)=O)ccc2ncccc2n1 66985,C(CC(=O)NCCCC(C)(F)F)(C(F)F)NC(CC(C)c1ccco1)=O 66986,C1(C)(C(N(CC(C)CNC(c2ccncc2C2CC2)=O)C)=O)CCCCC1(F)F 66987,C1(NC(=O)CNc2ccccn2)CCCN(C(c2cc(C3CC3)on2)=O)C1 66988,Cc1nccc(C(=O)NCCC2CC(F)(F)CN2C(=O)CC2CCOC2)c1C 66989,C(CC(=O)NC1(C)CC(NC(C2(O)CC2(C)C)=O)C1)(C(N)=O)NC(C)=O 66990,CC(CC(F)F)C(=O)N(CC(O)CNC(c1ccnc(CO)c1)=O)C 66991,N1(C(c2c(C)c(NC(C)C(C)C)ccc2)=O)CCC2CC(C)CCC2C1 66992,N1(CC(=O)NCC2(O)CN(C(C3CCC(=O)O3)=O)C2)CCCCCC1 66993,N1(C(CC(C)SC)=O)CCC2(CC1)CC(NC(c1sc(F)cc1Cl)=O)CO2 66994,C1(O)(C(C)NC(C(N2C(=O)CCC2=O)C)=O)CCN(C(=O)C2=CCC2)C1 66995,CC1CCN(C(c2conc2C(C)(C)C)=O)CCN1C(=O)CCc1ccccc1 66996,n1(CC)ncc(C(=O)NC(C)(C)C(=O)NC2CCCC2SC)c1C 66997,N1(C(c2c(CC)cc(N)cc2)=O)CC(NC(c2coc(Br)n2)=O)CC2(CCC2)C1 66998,n12nnnc1C2.c1(C2CCC2)ccccc1.c1(C2(N3CCC3)CC2)cccnn1 66999,CC(C)C(O)CNC(=O)C(C)(C)NC(c1ncn(C(C)C)n1)=O 67000,C1(C(=O)NCC(CCO)OC)(C(C)C)CCCN1C(C1CC(N=[N+]=[N-])C1)=O 67001,Cc1cnc2c(C(=O)NCC(CO)NC(=O)C(c3ccc(C)o3)C)c(C)nn2c1 67002,N1(C(c2cnc(OC)nc2C)=O)CCCC12CCN(C(=O)C(C)CF)C2 67003,c1(C(N2CC(C#C)C2)=O)cncc(CNC(=O)COCc2nc[nH]n2)c1 67004,c1(N2CC(C(C)NC(Cc3c(OC)cccc3)=O)C2)ncnc2c1CCC2 67005,C1(N(C(CCC)=O)C)CCCN(C(c2cnn(CCCOC)c2)=O)CC1 67006,CC(CC(F)F)C(=O)N1CC(N(C)C(C2CC2c2ccc(F)c(F)c2)=O)C1 67007,c1(C(=O)NCC=CCNC(c2cccc(C)c2)=O)ccc2nc(N(C)C)[nH]c2c1 67008,c1(OCC)c(F)cc(C(N2CCC(CN3CCN(C)CC3)C2)=O)cc1F 67009,CCCCCCN(CC(=O)NCCC1(NC(c2ccc[nH]2)=O)CCC1)C 67010,CN1CC2CC2(NC(=O)C(=O)NCCOC2CCCCC2)S1(=O)=O 67011,N1(C(C2(F)CCCC2)=O)CCC2(CC1)CN(c1ccnc3ncnn13)CCO2 67012,c1(NC(C2C(C(=O)OC)C2)=O)ccc(C(=O)Nc2cc(Cl)ncc2F)cc1C 67013,Cc1ccc(CN2CC(F)CC2C(=O)Nc2ccnc(-c3cccnc3)c2)cc1 67014,Cc1cnc(C(=O)NC2CCCCC2NC(=O)Cn2cnnn2)c(Br)c1 67015,C1(C)(C(=O)NCCCNC(C2(NC(C)C)CC2)=O)CCOC1 67016,n1(CC)ccc(C(=O)NCC2(NC(=O)C=CC(=O)NC3CC3)CCOC2)c1C 67017,C1(NC(C(CNC(=O)C=CCN2CCCC2)OC)=O)CCOCC1F 67018,c1(SCC2CC(C(C)OC)C2)cc(F)c(F)c(Cl)c1 67019,C1(OC)CC(CNC(=O)Cc2cc(C)cs2)(NC(C2CCCN2C)=O)C1 67020,N1(C(C2(S(C)(=O)=O)CC2)=O)CCC2(CC(NC(C3CCC=CO3)=O)C2)C1 67021,C1(CCCC)CN(C(=O)OC(C)(C)C)CCN1C(=O)Oc1ccnn1C 67022,c1(C(=O)NCCCCN(C(Cc2c(C)cco2)=O)C)sc(N2CCCC2)nc1Cl 67023,CCCCCCC(C)CC(=O)NC1CCN(C(c2cnc3n2CCC3)=O)C12CC2 67024,N1(C(c2c(CC)nccn2)=O)CCCC2(CCN(C(=O)C(C)NC(C)=O)CC2)C1 67025,C1(C(N2CCN(C(CC=C=C)=O)C(CO)C2)=O)CC12CCC1(CC2)OCCO1 67026,c1(OC)c(CNCC2CCCN2C(=O)CCC(N)=O)cc(F)cc1F 67027,CC1CC=C(C(=O)N2CCN(C3CN(C(C4C(C5CC5)C4(F)F)=O)C3)CC2)CC1 67028,C(=O)(C(C(C)(C)C)OC(C)(C)C)N(CC(C)NC(C12CC(C(C)(C)C)(C1)C2)=O)C 67029,N1(C(CN2CC(=O)NCCC2)=O)CC2CC(F)(F)CCC2(C(=O)O)C1 67030,C#Cc1cccc(C(=O)NCC2(F)CCN(C(=O)C(C)(C)CCOC)CC2)c1 67031,c1(C(N(CCCN(C)C(c2ccc([N+](=O)[O-])o2)=O)C)=O)cnc(N)c(N)c1 67032,C1(c2nc(-c3ccc(OCC)cc3)nn2CC2CCCO2)CC2C(C1)C2(F)F 67033,Cc1cc(C)n(CC(c2nc(C3CC34CC4)nn2-c2ccc(Cl)cc2)C)c(=O)n1 67034,Cc1nc(C#N)c(-n2cc(-c3ccn(C4CC4(F)F)n3)nn2)n1C 67035,c1(C(=O)NCC(COC)NC(=O)C(C)n2cccn2)conc1C1CCCC1 67036,N1(C(C2CCCS2)=O)CCC2C(C1)CN2C(=O)Cc1cccc(Cl)c1 67037,C1(NC(c2ccc(Br)o2)=O)CCC(CNC(c2cccn2C2CC2)=O)C1 67038,C1(O)(C(=O)NCC2(CCNC(C3(C)COCCO3)=O)CC2)CN2CCC1CC2 67039,C1(CC(=O)NCC(CC)NC(c2cc(C(N)=O)c[nH]2)=O)COc2ccccc2O1 67040,C1(C(=O)NC(Cc2ncn(C)c2)C(=O)O)CC12CCSCC2 67041,C1(NC(c2cc(C)c(Cl)s2)=O)C2CC1N(C(=O)C(O)Cc1cnc[nH]1)C2C 67042,c1(OC)c(C(=O)NCCC(C)N(C)C(c2cnn(C(C)(C)C)c2)=O)csc1C 67043,c1(C(=O)NC(CNC(C(COC)COC)=O)(C)C)cc2n(n1)CCCC2 67044,Cc1csc(C(N2CCOC(CN(C(=O)CN(CC(C)(C)C)C)C)C2)=O)c1Cl 67045,c1(CN(S(=O)(=O)c2cccs2)CCCN(C)C)cc2ccc(Cl)cc2[nH]1 67046,CCCCCC(CC)C(=O)N1CC(CNC(=O)Cc2nonc2C)C1 67047,N1(C(Cc2nc(C)[nH]n2)=O)CC2CC(NC(=O)Cc3cc(Cl)cc(Cl)c3)C(C2)C1 67048,C1(C)(CCNC(COCC(C)C)=O)CCN(C(=O)CSC(F)F)CC1 67049,CCC(C#N)C(=O)N1CC(C(=O)N(CCO)CCO)(COC)C1 67050,CCCC(CC)C(=O)NCC1CC2CC2N1C(c1cnn(CCOC)c1)=O 67051,O=C1CN(CCCCCC(N2CC(O)CC3(CCCC3)C2)=O)c2ccccc2N1 67052,c1(C(=O)NC2C(C)CN(C(=O)CC3CCNC3=O)C2)ccc2c(c1)C(C)CN2 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67088,C1(NC(c2cc(C)c(O)nn2)=O)CC1C1CCCN(C(=O)CCn2ccnc2)C1 67089,CC1(C(=O)NC2CC(CNC(=O)CSc3cccc(Cl)c3)C2)CCCCC1(F)F 67090,N1(c2nnc(CCC)s2)CC2CC(NC(c3ccn(C(CC)CC)n3)=O)CC1C2 67091,c1(C(=O)Nc2nc(-c3ccccc3C(F)(F)F)cs2)ccncc1Cl 67092,C(C(F)(F)C(F)F)N(C(C(C1CCC1)NC(c1ccccc1F)=O)=O)C1CC1 67093,C12(NC(=O)CCc3cncs3)CCCC1(F)CN(C(=O)Cc1cc[nH]n1)C2 67094,N1(C(C2(F)CCC(C)CC2)=O)CCOC2(C1)CN(C(C1(C)CCOCC1)=O)C2 67095,C(=O)(C1=NOC(C)C1)NCC1CC(NC(c2cccc(SCC#C)c2)=O)C1 67096,N1(C(CN(c2ccccc2)CC(=O)OCC)=O)CCCC(C)(C)C1CNC 67097,C1(CC)CC(C(=O)N(CC(CC)NC(=O)C=C(C)c2ccco2)C)CC(=O)N1 67098,N1(C(c2cc(SC)c(N)cc2)=O)CC2CCN(C(c3snnc3C(C)C)=O)C2C1 67099,c1(C(C)F)cccc(NC(C2CN(C(C3OC4CCC3C4)=O)CC2C)=O)c1 67100,c1(C(=O)OC)cc(C(=O)NC2CCCCC2NC(=O)CCS(C)=O)n(C)n1 67101,N1(C(C2CC=CC(NC(C3=CC(C)(C)C3)=O)C2)=O)CCCC(C2(C)CC2)C1 67102,C(C)(C(=O)N1CC(CNC(c2cocc2C)=O)CC(C)C1)(C(C)C)OC 67103,N1(C(Cc2c(C)nsc2)=O)CCN(C(c2nocc2Cl)=O)C2CC12 67104,C(=O)(C(CC1CC1)NC(C1(C(C)(F)F)CC1)=O)NC1C(N(C)C)CC1 67105,CCC(C)CC(C)C(=O)N1CC(NC(=O)CCOc2ccccc2Cl)C1 67106,C1(C(=O)Nc2ccc(C)cc2F)CN(C(c2cc(C#N)oc2C)=O)CC12CCC2 67107,c1(NC(C2CCN(Cc3scnc3Cl)CC2O)=O)cc(F)c(F)c(F)c1F 67108,N1(C(CCc2cccc(C)c2)=O)CCCCC(NC(c2nn(C)cc2Br)=O)C1 67109,C1(C(N(CC(=O)N(CC(=O)NC)C)C(C)C)=O)COCCN1C 67110,NS(=O)(=O)CCC(=O)NC1CCN(C(C2(F)CCCOC2)=O)C1 67111,C1(N(C(c2cnc(CCC)s2)=O)CC)CCN(C(=O)Cn2cncn2)CC1 67112,c1(NC(=O)CC2CC3CC(=O)C2C3)ccc2nccnc2c1I 67113,c1(CNC(C(C)NC(CC)=O)=O)n[nH]c2c1CN(C(C1CN(C)C(=O)N1)=O)CC2 67114,C1(C(=O)NCC(C)(CO)NC(CCS(=O)(=O)NC)=O)CCc2ccnn2C1 67115,CC1(C)CCCC(CC(=O)NC2(C)CCN(C(C3(O)CC3)=O)CC2)O1 67116,C1(C#N)(C(=O)NCCN(C(c2ccc(N(CCCC)C)cc2)=O)C)CCCOC1 67117,C1(NC(CCN(C(C(C=C)O)=O)C(C)C)=O)CCNC(=O)CC1 67118,N1(C(=O)CCc2cc[nH]n2)CCN(C(C23CCCC(C2)OC3)=O)CC1CCO 67119,c1(NC(C(CCNC(=O)CCCn2cncn2)O)=O)ccc(O)c(F)c1 67120,Nc1cc(Cl)cc(F)c1C(N1CC(CNC(=O)C=Cc2ccc(C(N)=O)o2)C1)=O 67121,c1(C(=O)NC(CNC(C2(CC#N)COC2)=O)CO)cc(Cl)cc(F)c1Br 67122,S(=O)(=O)(c1cncn1C)N(C)Cc1ncco1 67123,C1(NC(C2C(=O)NCCC2)=O)CCC(O)CN(C(=O)CCCc2ccccn2)C1 67124,C1(NC(CC(=O)NCC#C)=O)CS(=O)(=O)CC1NC(c1nccc(N)c1Cl)=O 67125,c1(C(=O)NCC2C(NC(CCCN(C(C)=O)C)=O)C2)c(Cl)nsc1Cl 67126,C(=O)(C(O)CCC(C)C)N1CC2C(NC(c3ccc(OC)c(C4CC4)c3)=O)(C2)C1 67127,c1(NCCN(C(=O)CC2CCCCC2(F)F)CC)ncn(C)c(=O)c1Br 67128,c1(C(=O)NCCCCN(C(=O)COc2ccccn2)C)cc(-c2ccco2)on1 67129,C=C(CC)CN=C(NCc1ccc2c(c1)CNC2=O)NCC1CCCCO1 67130,C1(C(C(=O)NCC=C)N(C)Cc2ccc(C)cn2)CCCC(CC)C1 67131,C(C(CC(=O)Nc1cnn(C(C)C)c1)NC(c1coc(C(C)C)n1)=O)OC 67132,O=C1CN(CC(N2CCN(C(c3nc(CC4OCCO4)ns3)=O)CC2)=O)CCCN1 67133,c1(C(=O)NCC(CC(C)C)NC(=O)C(O)c2ccsc2)csc2ccc(F)cc12 67134,C(=O)(C#CC(C)(C)C(F)F)N(C)CCNC(C1CCCN1c1nccs1)=O 67135,C1(NC(C(C)Cc2cnn(C)c2)=O)CN(C(c2sc(N(C)C)nc2Cl)=O)CC1O 67136,Cc1ncc(Cl)c(C(=O)NCC2CCN2C(=O)Cc2nnn(C(C)(C)C)n2)n1 67137,N1(CC(=O)NCC2CCN(C(=O)Cc3cnn[nH]3)C2)CCC(n2cccc2)CC1 67138,C1(CC)CCN(C(=O)Cc2ccsc2C)C(C(=O)N(CC(O)C2CC2)C)C1 67139,C(C1C(C(=O)NCCC(C)N(C)C(C2CCC=CO2)=O)C1(C)C)=C(C)C 67140,C(=O)(C(CCc1ccc(Cl)cc1)N1CCC(O)(C(N)=O)C1)NCCCSC 67141,C=C(C)c1cncc(C(=O)NCCSCCC)c1.C(C)(=O)O 67142,N1(C(C(C)c2ccco2)=O)CCCC(NC(c2ncc(Cl)nc2Cl)=O)C1C 67143,Cc1ncnc(C)c1C(N1CCCC(C(=O)NCC(C)(O)C2(C)CC2)C1)=O 67144,c1(-n2cc(C3OCCN(C(CCC4CCC(C)O4)=O)C3)nn2)cc(F)cnc1Br 67145,N1(C(C2C(CNC(CCCC(CC)C)=O)CCO2)=O)CCc2ncn(C)c2C1 67146,c1(CC)noc(C)c1NC(=O)COC1CC(NC(C2(C#N)CC2C)=O)C1 67147,c1(CCNC(C(C)SC)=O)ccc(CNC(=O)C(N2CCSCC2)C)cc1 67148,Cc1cccc(Cl)c1CC(N1CC2C(N(C(=O)COC3CCCC3)C)C2C1)=O 67149,C12CNC(=O)CN1C(=O)C(C1CCCC1)NC2=O.C1(CC)(CO)CCCC1 67150,CCC(CC(=O)NCC1(OC)CCN(C(c2nn(C)nc2Br)=O)C1)SC 67151,C1(NC(C(C)OCC(C)C)=O)CCCC(CNC(c2cnc[nH]c2=N)=O)C1 67152,c1(C(N2CC(C)C(NC(C3CCCC(CF)C3)=O)C2)=O)nn(C)c(Cl)c1Cl 67153,N#Cc1ccc(CC(C#N)C(=O)Nc2cccc(F)c2)cc1 67154,Cn1c(NC(=O)CC(O)c2ccccc2)nc2cc(Br)c(Cl)cc12 67155,C(C(=O)NCCC1CCN(C(=O)C(C)N(C)C)C1)(C(C)C)NC(C)=O 67156,CCC(CCOC)C(=O)NC(C)CCCC(=O)N1CC(F)(C2CC2)C1 67157,N1(C(CCCN(C(=O)OC)C)=O)CCN(C(=O)CCc2ccc(C)cc2)C2CC12 67158,c1(CC(=O)N(CC(C)(C)CNC(=O)C=C2CCC2)C)ccccc1O 67159,C#Cc1ccc(C(=O)NCC2CC2CNC(C2CC(C)(F)C2)=O)c(F)c1 67160,C(c1ccc(=N)[nH]c1C)=CC(N1CC(COC)(NC(=O)CC(C)C)C1)=O 67161,CC1(C(=O)NCc2cc(C(=O)NCCCC3(O)CCC3)on2)CCOC1 67162,C1(C(=O)NCC(CC)NC(c2scnc2C)=O)CCCNS1(=O)=O 67163,N1(C(C(C=C)(C)CC)=O)CC2CC(NC(c3ccc(Cl)cc3Cl)=O)C(C2)C1 67164,N1(C(COC(C)C)=O)CC2CCCC1(CNC(c1coc3ccccc13)=O)C2 67165,C(=O)(C#CC1(C)CCCO1)NC.C1(NC(CN(CCC)C)=O)CCCC1C 67166,C1(NC(C2CCC(CC)O2)=O)CC2CCC1(C(N1CCC1c1ccccc1)=O)C2 67167,C1(CNC(c2c(C)oc(CO)c2)=O)CC2(CCN(C(C3(C)CC3(F)F)=O)C2)CO1 67168,c1(C(=O)NCC2N(C(C3C(C)C3C)=O)CC(C)(C)OC2)c(F)cc(F)c(F)c1F 67169,c1(C(=O)NC(CNC(c2cc(C(C)C)on2)=O)(C)C)ccc(F)c(N)c1F 67170,C1(NC(c2cc(Br)co2)=O)CN(C(=O)CC2CSC2)CC2(CC2)C1 67171,c1(C(=O)NCC23CCCC2CN(C(c2cnns2)=O)C3)cnn2c1C(=O)NCC2 67172,N1(C(Cc2cc(OC)c(F)cc2)=O)CC2CCC1CC2NC(=O)CC(C)(C)C 67173,O(N1CCC(NC(C2CSCCN2C(=O)C(C)S(C)(=O)=O)=O)CC1)CC 67174,CC1CCC(NC(=O)CC2COCCOC2)CN1C(c1cc(C(N)=O)ccn1)=O 67175,c1(CCC(=O)N(C2CN(C(=O)CC3(CO)CCCC3)C2)C)ccc(F)cc1 67176,N1(C(c2cc(C(C)=O)[nH]n2)=O)CCOC2CN(Cc3c(C)cc(Br)cc3C)CC12 67177,CC1(C)C(=O)NC2CCC(C(=O)Nc3ccc(SCc4nc[nH]n4)cc3)CC12 67178,C1(CNC(=O)OC(C)(C)C)CCN(C(=O)Nc2cn(C)cc2C(F)(F)F)C12CC2 67179,c1(CS(C)(=O)=O)ccc(CN(C)C(C2CCN(C(CC(C)O)=O)C2)=O)cc1 67180,C1(OC)(OC)CC(C)(C(=O)N(C)CC2(O)CN(C(c3n[nH]c(C)c3Cl)=O)C2)C1 67181,CCS(=O)(=O)c1ccc(Cl)c(C(N2CCC(N(C(=O)C(C)C#N)C)C2)=O)c1Cl 67182,c1(CC(=O)NC2C(NC(CC3CC(SC)C3)=O)CCC2)ccc(C)cc1 67183,N1(C(c2nn(C)c(=O)cc2)=O)CC2(CCC2)CC1CNC(=O)C(F)C1CCOC1 67184,S(=O)(=O)(c1ccc(C#N)c(N(C)CCF)c1)N(C1C(C)CCC1)C 67185,C1(CNC(CCSC)=O)CN(C(=O)CC2CCCOCC2)CCC12CCOC2 67186,C1(NC(CCC(C)OC)=O)CN(C(=O)CCn2nc(C)cc2C)CC2CC12 67187,C1(NC(Cc2c(C)n(C)nc2)=O)CCCN(C(c2cc[n+]([O-])cc2)=O)C1C 67188,c1(C(=O)NC2CCC(C)N(Cc3ccccc3)C2)cc(N)cc(O)c1Br 67189,N1(C(C(c2ccoc2)SCC)=O)CCCC(C(=O)NCc2nnc(O)o2)C1 67190,N1(C(c2c(CC)csc2)=O)CC(NC(c2cnc(C)s2)=O)C2CC12 67191,c1(C(=O)NCC2(F)CN(C(=O)CCC3CC(F)(F)C3)C2)cncc([N+](=O)[O-])c1 67192,CN1C(=O)CN(C(=O)CC2C3CN(C(C4CC(C)(C)CN4C)=O)CC23)CC1=O 67193,c1(C(N(CCNC(=O)C=CC2(C)CCOCC2)CC)=O)ccc2ncncc2c1 67194,C(=O)(CC(C)C(=O)OC)NCCN(C(C1CC1c1cc(F)ccc1F)=O)CC 67195,C1(O)(CC2(NC(C3(CC=C)CC3)=O)CCC2)CN(C(=O)C(C)OCC(C)(C)C)C1 67196,C(=O)(C(C(C)(C)NC)c1ccccc1)NC1C(CC)CN(C(=O)OC(C)(C)C)C1 67197,c1(CC)[nH]c(=N)sc1C(=O)NCC(O)CN(C)C(c1ccno1)=O 67198,c1(C(C)C(=O)NC2CCCN(C(=O)C=CCO)C2)ccc(S(=O)(=O)N(C)C)cc1 67199,N1(C(CCc2ccc(C)o2)=O)CC(C(N2CCC(CCF)CC2)=O)CC(C)C1 67200,c1(SCCC(=O)NCC(CC)NC(=O)C(C)SC)ccc(C)cc1 67201,Cc1c(Br)ccc(NC(=O)C(=O)N(CC(C)O)C(C)C)c1I 67202,Cc1cc2cc(C(=O)NCC(C)NC(C3(CO)CCCCC3)=O)c(Cl)cc2[nH]1 67203,C1(C(=O)NC2CCC(C(=O)NCC(C)CC3CCC3)C2)(OC)CCOC1 67204,C(=O)(CC1CC(C)(OC)C(=O)N1)N1C(CCC#C)CCC1.OC 67205,N1(C(COCCCCC)=O)CC2(C1)C(NC(c1cc(C)oc1C)=O)CCS2(=O)=O 67206,C1(C)(C(=O)NCCCOC(=O)NC)CCN(C(=O)C=Cc2cn(C)cn2)CC1 67207,Cc1nc2sc1C(=O)NC2.C1(C(=O)Nc2nccs2)CCOC(C)C1 67208,N1(C(C2Cc3cc(F)ccc3O2)=O)CCCCC2(C1)CN(C(c1cc[nH]c1)=O)C2 67209,C1(COC)C=CCCN1C(=O)COC1CCN(C(C2(CO)CCC2)=O)C1 67210,c1(C(CNC(C)=O)NC(c2c[nH]nc2[N+](=O)[O-])=O)ccc2ccccc2c1 67211,N1(C(C(C)SC)=O)CC(NC(=O)C=CCCC(C)C)CCC1C 67212,c1(NC2(C(=O)OC)CCOC2)ccccc1C.C1(CC2CCC2)C(=O)N1C1CC1 67213,Cc1nc2cccc(C(=O)NC3COCC3CNC(C34CCC(C3)C4)=O)c2[nH]1 67214,c1(CN(C)C(C2(F)CCN(C(c3cnc(Cl)nc3)=O)C2)=O)ccc(F)cc1 67215,c1(NCCCC(=O)OCc2nc(SC)nc(O)c2)ccc2c(c1)CCO2 67216,C1(F)(CNC(CCN(C2CC2)CC)=O)CCN(C(=O)Cc2nocc2C)C1 67217,C1(CC(=O)NCC2N(C(C(F)=CCC)=O)CCC2)COC2CC1C2 67218,c1(OC)c(NC(C2CCCN(C(C3CC3C)=O)C2)C)ncnc1Cl 67219,N1(C(CC)=O)CCC2(CC1)CC(CNC(=O)CC(O)CN(C)C)CO2 67220,S(=O)(=O)(CCCCCl)C1C(C(=O)NC(C2CCCCC2)CO)C1 67221,C12(C(=O)NCC3C(C)CCN(C(C4(O)CCCCC4)=O)C3)CCC(CC1)C2(C)C 67222,C=C1Cn2c(C(=O)NCC3CC4CN(C(=O)C=CSC)CC34)nnc2S1 67223,C1(NC(C2(SC)CCC2)=O)COC2(CCN(C(c3ocnc3C(F)F)=O)CC2)C1 67224,N1(C(Cn2c(C)c(Cl)cn2)=O)CC(C)N(C(=O)CC(F)(F)C(C)C)CC1C 67225,CC1C(NC(=O)CN(CC(C)(C)C)C)CCCN1c1ccc(C(F)(F)F)cn1 67226,N1(C(CC(=O)OCC)=O)CC2(CC(CC(=O)NCC3(C#N)CC3)C2)C1 67227,N(C(=NCCCCC(F)(F)F)NCCC1(O)CCCC1)C(CC)CC 67228,C1(CNC(c2nnnn2-c2ccccc2)(CC)C)CC(C2CC2)=NO1 67229,Cc1cc(NC(C2CC(C)(C)CN2C(C2CCCO2)=O)=O)ccc1O 67230,c1(OCC=C)ccc(Cl)c(NC(C2CCN2CC2CCCC2)=O)n1 67231,N(C1CN(C(=O)C2=CCCOC2)Cc2ccccc21)C(Cn1c(C)nnn1)=O 67232,CC1CCCC(CC(=O)NCC(C2CCCCC2)NC(C2CC(F)C2)=O)C1 67233,CC(C(=O)N1CC2CC1C2NC(c1ccc(F)c(C(F)F)c1)=O)C(F)(F)F 67234,c1(N2CCC(CNC(C(COC)(C)C)=O)C2(C)C)cc(C#N)nc(C2CC2)n1 67235,c1(C(N2CCN(C(C(CC)OC)=O)C(C3CC3)C2)=O)cc2ccc(F)c(F)c2o1 67236,C1(c2cn(C(C)(C)C)nc2)CN(C(=O)C(c2cnn(C3CC3)c2Cl)=O)CCO1 67237,C1(NC(CC(C)(C)N(C(c2c(C)coc2)=O)C)=O)CN(C)CC1(F)F 67238,C(=O)(CCN(C(C1CC1Cl)=O)C(C)C)NCC1C(C(=O)OC)C1 67239,C1(CCC)CN(C(c2cnc(=N)[nH]c2)=O)CC1C(=O)NC1(C)CCSC1 67240,C1(COC)(NC(c2coc(C3CCC3)n2)=O)CCN(C(C2COC2)=O)C1 67241,Cc1cccnc1C(C(C)(C)C)NC(=O)NCC1(OCCO)CCC1 67242,C(C)(CCCC(=O)NCCCCn1ccnc1)NC(Cc1c(C)scc1)=O 67243,C1(NC(C2(C)CCCCCC2)c2n(CCOCC)nnn2)CCCC(C)(C)C1 67244,N1(C(CNC(CCC(C)C)=O)=O)CCC(NC(=O)CC2CNC(=O)C2)C12CCC2 67245,c1(C(N(CC(N2CCCC2CNC(c2ccco2)=O)=O)C)=O)c(N)cccc1Cl 67246,N1(C(C(=O)NC(COCC)C)=O)CC2CC2C2CC12 67247,c1(C(=O)NC2CC(CNC(C3CCCC3(F)F)=O)C2)ccc2nc(S)oc2c1 67248,C1(C(N(CC(CCC)O)C)=O)CCN(C(=O)C#CC2(C)COC2)C12CCC2 67249,C1(=CC(=O)NCC(CN(C(C(CC)O)=O)C)O)CC2CCC(C1)N2C 67250,N(C(=NCCCN(S(C)(=O)=O)C)NCC1CCCCO1)C(CC)C 67251,CC1=C(C(=O)NC2CC3CC(NC(C4CC(C(C)C)=NO4)=O)CC3C2)CCCC1 67252,CC1CCCN(C(c2c(NCCC3(C)CCCO3)cccc2)=O)C1 67253,c1(C(N2CCCN(C(c3cnc(C)o3)=O)CC2)=O)c[nH]c(C)c(Cl)c1=O 67254,Cc1c(C(N2CC3(CC3)CC2CNC(=O)CNC(N)=O)=O)sc2ccccc12 67255,C(CC(C(=O)N1CC(O)C(O)C1)NC(C1SCC=C1C)=O)SC 67256,c1(C(CC)NC(C)C(=O)NC(C)C)nc(C(F)(F)F)n[nH]1 67257,C1(C)(CNC(CC2C=NN(C)C2=O)=O)CN(c2cc(C(F)(F)F)ncn2)CCO1 67258,CC1CCN(C(=O)CCc2c(Cl)cncc2Cl)CC1NC(=O)C=CC1CC1 67259,c1(C(=O)NC(C2CC2C(=O)N(C2CCCC2(C)O)C)C)ccnc(O)c1F 67260,C1(CNC(C(C)OC)=O)CCCC1NC(C1CCC2CC12)=O 67261,c1(C(=O)NCC23CCC(CC2)N(C(C2CC2(Cl)Cl)=O)C3)ccc(F)cc1[N+](=O)[O-] 67262,c1(C(=O)NC(C(C)NC(CC(C)C)=O)C)cc2c(cc1[N+](=O)[O-])OCCCO2 67263,C1(CNC(CC=CC)=O)CC(NC(c2cn(C)cn2)=O)C12CCC2 67264,N1(C(C2CCOCC2)=O)CCC(NC(C2(C3CCCO3)CC2)C2CC2)C(F)C1 67265,C(=O)(CC1C(=O)Nc2ccc(Cl)cc21)NC1CC(C)(NC(CC(=O)N(C)C)=O)C1 67266,N1(c2nnc(C(C)(C)C)s2)CCCC2(CC(NC(=O)Cc3ccc(O)nc3)C2)C1 67267,C1(NC(c2ccc(I)c(Br)c2)=O)CN(C(=O)Cn2cc(Cl)cn2)CC1(F)F 67268,c1(CN(CCC)C(=O)Nc2nc(C(C)C)ns2)cc(Cl)ccc1Br 67269,C(=O)(C(F)C(CC)CC)N1CCN(CC(C)NC(c2nc(CC)oc2)=O)CC1 67270,C(=O)(C1=CS(=O)(=O)CCC1)NC(c1cccc(O)c1)C(=O)OC 67271,n1(CC)cnc2nc(N3CCN(C)C4(CCC4)C3)nc(N(CC(F)(F)Br)C)c12 67272,CCC(CC(C)CO)NC(=O)N(C1CCSC1)C 67273,CCS(=O)(=O)CC(=O)N(C(C)CCNC(=O)CCCC(C)c1ccccc1)C 67274,CCC(CNC(=O)CC1CCCC1NC(=O)CCC(=O)NC)C(C)C 67275,C1(CNC(C(C)(O)CCc2ccccc2)=O)CC2CCC1N(C(=O)CCCF)C2 67276,C1(NC(=O)OC(C)(C)C)CCCN(CCNCc2ccc(O)c(O)c2)CC1 67277,C1(CNC(C(C2CCN(C(CNC(=O)NC)=O)C2)F)=O)(CO)CCN(C)C1 67278,c1(C(=O)NC2C(C)(C)CN(C(c3occc3C3CC3)=O)C2)ccnc2c1CCN2 67279,C(=O)(CN=c1[nH]c(C)cs1)NCC1CN(C(c2cnc(OC)c(C)c2)=O)CC1C 67280,N1(C2CN(C(C=CC(C)NC(c3ccco3)=O)=O)C2)CCCS1(=O)=O 67281,c1(N(C(C)=O)C(C2CCOC2C)=O)ccc(-c2cnco2)cc1Cl 67282,C1(CCC)CN(C(=O)CC(C)C)CC1C(=O)NCC(C)(O)C1CCC1 67283,C1(C(C)C)CN(C(=O)CC(C)c2cnn(C)c2)CCN1C(c1ccoc1Cl)=O 67284,C1(CCCOC(C)C(=O)NCCc2ccccc2)CCCN1C(=O)CC1(C)CC1 67285,C(=O)(C(F)C(F)(F)F)NCC(C)N(C)C(c1ccc(CO)cc1F)=O 67286,CN1CCC(C(=O)NC2(CNC(C3CCC(F)C3)=O)CCC2)CC1=O 67287,N1(C(C(COCC)n2cc(C(OCC)OCC)nn2)=O)CC(C#N)CC1C 67288,C(c1ccc(F)nc1)=CC(=O)NC(CNC(c1c(C)nc(N(C)C)s1)=O)C 67289,C1(N(C(c2ccc(CNC(C)=O)s2)=O)C)CCCN(C(C2COC(=O)O2)=O)CC1 67290,C(=O)(CC(C)(C)CNC(c1cc(Cl)n[nH]1)=O)NCC(C)Cc1cn[nH]c1 67291,C(=O)(C(C)(O)C(F)(F)F)N1CC(CNC(C2CC(OC)C(OC)C2)=O)C1 67292,C(CCC(CCC)NC(c1n[nH]c(C)c1C)=O)NC(c1cn(CCCC)nn1)=O 67293,C1(CNC(C(C)SCC)=O)(CO)CCCN(C(C2CCCN2C(C)=O)=O)C1 67294,C(=O)(CC1=CCOCC1)N1CC(C(=O)Nc2cc(C)c(O)cc2)C(C)(C)C1 67295,Cn1ccc(=O)c(C(=O)NCCCN2CCN(C(C3CCS(=O)(=O)C3)=O)CC2)c1 67296,Cc1cc2ccccc2nc1C(N1CC2CCN(C(c3csnn3)=O)CC2C1)=O 67297,C(CCCCC(=O)N1CC(NC(=O)CSC)CC(C)C1)OCC 67298,c1(C(N)=O)cc2n(n1)CCCN(C(=O)CCCCCl)C2 67299,CC1(C)CC(CC(=O)NC(CNC(C2(CO)CCCO2)=O)C2CC2)CO1 67300,N1(C(CCS(=O)(=O)NC)=O)CCC2(CC1)CC2NC(=O)C(c1cccc(C)c1)C 67301,c1(C(=O)OC)cc(NC(c2sc(NC(C3CCCS3)=O)nc2C)=O)c(C)cc1Br 67302,c1(C(N2CC(C)OC(CCNC(=O)C3=CCCC3)C2)=O)cc(C#N)ccc1F 67303,c1(C(=O)NCC2CCN(C(CC3ON=C(CC)C3)=O)C2)cc(C)nc2ccnn12 67304,N1(C(c2c(C)nco2)=O)CCCC(O)(CN(C(=O)C(C)CN2CCCCC2)C)C1 67305,C1(NC(=O)CN(C(=O)CC2CSC2)C2CC2)CN2CCCC1C2 67306,CC(CN1CCOCC1)N=c1[nH]c(=NC(C)c2nc[nH]n2)[nH]c2c1CCCCC2 67307,Cn1ccc(-n2cc(C(CC(N)=O)NC(=O)CC3CCCSC3)nn2)cc1=O 67308,C1(C(=O)NCC(CC)NC(=O)CCn2cc(C(=O)OC)cn2)CCOC1C 67309,c1(C(=O)Nc2cc(Br)cc(I)c2)cccn2c(-c3ccc(O)c(CO)c3)cnc12 67310,n1(CCCOC(C(C=C)C)=O)nc(O)c2ccccc2c1=O 67311,c1(CN2CC3CN(C(=O)CCc4ccccn4)CC32)ccc(I)c(F)c1F 67312,C(=O)(C#CC1CCCOC1)NCCOCCN(C(CC(C(=O)OC)C)=O)C 67313,CCC(C)C(C)(O)CNC(=O)C(CC(C)C)ONC(C1CC12CC(OC)C2)=O 67314,N1(CCN(C(CN(C(=O)C(C)N(CC)CC)CCC)=O)CC)CCCCC1 67315,CC1CCCC(O)(CNC(C2CC(n3cc(CC4CCOC4)nn3)C2)=O)C1 67316,N1(C(CCCN(C(C(CCC)C)=O)C)=O)CCCC(C)(CCC)C1 67317,c1(CNC(C(CO)OC)=O)ncccc1C(=O)N(CCCCSC)N(C)C 67318,N1(C(c2c(CC)ocn2)=O)CC(NC(c2cc(O)ncn2)=O)C2CCCCC12 67319,Cc1ccc(Cl)c(C(=O)NCC2(O)CCN(C(C3CC34CCCC4)=O)CC2)c1N 67320,C1(OC)CC(CCNC(=O)CC(C)(C)C)N(C(=O)CCn2cncn2)C1 67321,CCCC(O)C(CO)NC(C12CC1CCN2C(C1CCCC(=O)CC1)=O)=O 67322,C(=O)(C(F)C(C)(C)O)NCC(C1CCN(C(=O)CCOCC(C)(C)C)CC1)C 67323,N1(CCC)CCCCC1C(=O)N(C)CCC1CCCCN1C(c1cnc(C)s1)=O 67324,N(C(=NCc1cccs1)NC1CC12CCCC2)CC(F)F 67325,CCCC(CCO)NC(=O)CC1(N(C(=O)C(CC)OC)C)CC1 67326,c1(OC)cc(C(=O)NCCc2ccccc2O)cc(C)c1 67327,c1(N(C(C(=O)NC2CCC(OCC(=O)O)CC2)=O)CC2CC2)ccc(Cl)cc1Cl 67328,C12(CNC(C(C(C)O)C)=O)CC(NC(=O)CC3CC3)(C1)C1(CCOCC1)O2 67329,N#Cc1cc(C(N2CCC(F)(C(=O)N(C3CCOCC3)C3CC3)C2)=O)cs1 67330,C1(NC(=O)C=C2CCCCC2)(CF)CCN(C(=O)C(c2cccc(F)c2)F)C1 67331,N1(C(C2(CCCC)CC2)=O)CCCC(C2CCCN(C(C3C4COCC34)=O)C2)C1 67332,N1(C(CP(C)(C)=O)=O)CCOCC(NC(c2ccccc2Cl)=O)C1 67333,N(C(=NCCN1CCOC1=O)NCC1CCCCO1)C1CC(C)OC1 67334,CS(=O)(=O)c1cnn(CC(=O)NC2CCCC(NC(=O)CSC(F)(F)F)CC2)c1 67335,c1(CC(=O)Nc2nc(C(C)NC(C)=O)oc2)cncc(Cl)n1 67336,C1(NC(C(C)NC(CC)(C)C)=O)CC(C)(C(=O)NCC(F)(F)F)C1 67337,Cc1cc(CO)cc(CC(N2CCC2Cn2cc(C3CCCC3O)nn2)=O)c1 67338,CCCC(CC)CC(=O)N1CC2CCC(C1)N2c1nc(Cl)nc(C)c1F 67339,C1(CNC(C2(OCC)CC2)=O)CN(C(=O)C(C)C(F)F)CC1(F)F 67340,N1(C(C2C(C)(Br)C2)=O)CC23CCCCC2(C1)CN(C(C1CCCC(O)C1)=O)C3 67341,C1(Nc2nccc(OC)n2)CN(C(c2cnccc2Cl)=O)CCC1C(F)(F)F 67342,C1(COC)CC(CNC(C2CC2C(C)(C)C)=O)N(C(=O)COCC(C)C)C1 67343,c1(CN(C)C(C23COCC(C2)C3)=O)ccccc1CNC(C1(F)CC=CCC1)=O 67344,c1(C(N2CCC(CNC(c3on(C)c(=O)c3)=O)C23CC3)=O)nnn2c1COCC2 67345,C(=O)(C(C)(C)C(C)(C)C)NC1CN(C(CC2C(C(=O)OCC)C2)=O)C1 67346,Nc1ncc(C(N2CC(CNC(c3ccco3)=O)C2)=O)cc1Br 67347,c1(C(=O)NC(CNC(CC2CC(=C)C2)=O)C2CC2)nccc(N)c1Cl 67348,c1(C(N2CCN(C(C3CC(=O)C3)=O)CC2C(F)F)=O)cc(F)cc2nccnc12 67349,Cc1c(C(=O)N(C)CC2CCN(C(=O)C(F)CC3CCOC3)CC2)cncc1F 67350,C1(C(=O)NCC2CC(OC)C2)(NC(=O)CCC2(C#N)CCC2)CCSC1 67351,C(=O)(C(C)(C)C(=O)NC(C1CCCCN1C(c1cc(Cl)n(C)n1)=O)C)OCC 67352,C1(CNC(c2ccc(OC)o2)=O)CCC(CNC(=O)C(O)C2CC2)CC1 67353,Cc1cc(Cl)c(Cl)cc1C(N1CCCCC1CNC(c1cn(C2CC2)nn1)=O)=O 67354,C1(C(N2CCC(N(C(=O)CC(C)(C)C3CC3)CCC)CC2)=O)CC(C2CCC2)C1 67355,c1(N(c2ncc(I)cn2)C)cc(-c2nc(=N)[nH][nH]2)cc([N+](=O)[O-])c1Br 67356,Cc1[nH]c2ccccc2c1C(N1CCC2(C1)CN(C(C1C(F)(F)C13CC3)=O)C2)=O 67357,C=CCC(C(=O)N1CC(CCNC(c2cc(Br)cnc2C)=O)(OC)C1)C(C)C 67358,c1(CNC2CN(C(CCc3c(C)noc3C)=O)CC2C)cc(F)cc(C#N)c1 67359,c1(N(CCNC(C2CC2C(=O)OC)=O)CC)cc(C(C)C)nc(C)n1 67360,N1(C(C(C)N2CCCC2)=O)CCCCC(CNC(=O)CN(c2ncccn2)C)C1 67361,N1(C(CC=C)=O)CC(CN(C)C(c2cc(Br)ccc2C)=O)C2(CC2)C1 67362,C1(N(C(c2cc(OC)ns2)=O)C)CCN(C(c2cccc(C)c2O)=O)CC12CC2 67363,C1(CNC(C2(OCC)CCOC2)=O)(CNC(=O)CC(F)F)CC12CCC2 67364,C(CCC(C)(C)C(=O)NC(C1(O)CCC1)C)NC(c1c(=O)cc(C)[nH]c1)=O 67365,N1(C(CC2CC(C(=O)OC)C2)=O)CCCC(N(C(=O)C=CSC)C)C1 67366,c1(NC(=O)Nc2ccccc2)ccccc1OC1CC(c2nccc(CO)n2)C1 67367,CC(C)CCC(C(=O)NCc1ccnc(F)c1F)NC(c1cnn[nH]1)=O 67368,CC1CN(C(C2(Cl)CC2(F)F)=O)CC1NC(c1cc(CC(F)(F)F)nn1C)=O 67369,c1(C(=O)NC2CCN(C(C3CC(C#N)C3)=O)CC2O)cccc2c1OCCO2 67370,N1(C(CCOC(C)C)=O)CCC2CCN(C(c3cc(C(F)(F)F)n(C)n3)=O)C2C1 67371,c1(CNC(=O)Cc2cccc(C3CC3)c2)ncc([N+](=O)[O-])cn1 67372,c1(OC)cccc(CN2CCC(CNC(c3csc(C)n3)=O)C2)n1 67373,c1(C(=O)NCC(C)(C2CC2)NC(=O)CCNC(=O)C=CCl)ccc(CCF)cc1 67374,n1(CC(N2CCC(C(C)NC(C3CC(N=[N+]=[N-])C3)=O)CC2)=O)ncc(O)nc1=O 67375,C(CCN(C)C(c1ccc(OC)o1)=O)(C(C)C)NC(c1cc(SCC)on1)=O 67376,Cc1csc2ccc(C(=O)NC(C)CCCNC(C3CCC(O)C3)=O)cc12 67377,C(N=c1cc[nH]cc1S(=O)(=O)NCC1(C(N)=O)CCC1)C1(C)CC2CCC1C2 67378,C1(C(=O)NC23C(CN(C(C4(CC=C)CCC4)=O)C2)C3)COc2ccc(F)cc2C1 67379,C1(C(=O)NCC2(C(=O)NCCCOCC)CC2)CC=CCC1 67380,C(CC(C(C)(C)C)NC(C1CC(CF)C1)=O)N(C)C(c1ccnc(C(F)F)c1)=O 67381,N1(C(C2C=C(C)CS2)=O)CC2(C)CC1(C(=O)N(C1CCN(C(C)C)C1)C)C2 67382,Cc1ccc(C(N)=O)cc1C(=O)NCC1CC(NC(=O)C(C)CC(N)=O)C1 67383,Cc1nc(CCC(N2CCC(CF)(NC(=O)CC3CC34CC4)C2)=O)oc1C 67384,C#Cc1ccc(C(=O)NCCC(CNC(=O)CN2CCC(=O)CC2)OC)cc1 67385,C1(C(=O)NCC=CC)CCC(n2cc(CC(c3ccccn3)C)nn2)CC1 67386,Cc1cc(F)c(F)cc1C(N1CC2CC2(C(=O)Nc2ncc(Br)nc2Cl)C1)=O 67387,c1(CN2CC(C(=O)NCc3c(C)cccc3)SCC2)cc([N+](=O)[O-])cc(O)c1O 67388,C1(CC)CN(C(=O)Cc2cccnc2)CCC1NC(c1sncc1C)=O 67389,N1(C(c2cc(S(=O)(=O)NC)oc2)=O)CCOC2(C1)CN(C(=O)C(C)CC1CC1)C2 67390,c1(C(N(CC(O)CN(C)C(C2CCCN2N=O)=O)C)=O)ccn(C)c(=O)c1O 67391,C1(CC(=O)NCC(CO)NC(=O)CNc2ccccc2)CCCCCC1 67392,Cc1cccc(CN2CCC(F)(C(=O)Nc3ncc(Br)cc3Cl)C2)c1F 67393,C1(C(=O)OCC)CC2(CCCN2C(=O)NC(C(F)F)C2CCC2)C1 67394,N1(C(CCN(C)CC)=O)CCC2(CCCCN(C(C3(Cl)CC3(C)C)=O)C2)C1 67395,N1(C(N=c2nc(C)[nH]n2C)=O)CC(C)(C)OC2(CCOC2)C1 67396,c1(C(N2CC3CN(C(C(C)(C)C(F)F)=O)CC3C2)=O)nc2ccc(Cl)nn2n1 67397,N1(C(C2N(C)CC2)=O)CC2CS(=O)(=O)CC2(NC(c2ccc([N+](=O)[O-])cc2)=O)C1 67398,N1(C(C2C(C)OCC2)=O)C2CCC1CN(C(=O)Cc1ccnn1C)C2 67399,c1(OC)c(C(=O)NC2(C)CN(C(C3(C)CC3(F)F)=O)C2)ccnc1Cl 67400,C1(NC(Cn2c(C)nnn2)=O)CC2CC(C1)N(C(=O)CC1CC(F)(F)C1)C2 67401,Cc1cc(C(F)(F)C(=O)N(CC(C)NC(C2(O)COC2)=O)C)cc(C)c1 67402,C1(C(=O)NCc2cc(C(N(CC(C(C)C)OC)C)=O)n(C)n2)CCC(N=[N+]=[N-])C1 67403,c1(C(=O)NCCC2(O)CCN(C(=O)CN3CCOCC3)C2)nccc2nn[nH]c12 67404,c1(NC(C2CSCCN2Cc2ccc(Br)s2)=O)cnc(Br)nc1 67405,c1(C(=O)NC2(CCNC(CCc3cn(C)nc3)=O)CC2)cnc2[nH]ccc2n1 67406,C(CN=C(NCCOc1ccccc1)NCc1cnccn1)C1CC(F)C1 67407,C1(C(=O)NC)CN(C(=O)CC2CCC(NC(=O)CCC(C)OC)C2)CCO1 67408,CC(C)C(C)C(CNC(=O)COCCF)NC(c1cc(C#N)on1)=O 67409,c1(NC)cccc(C(=O)NCCCCOC)n1.N12CC(O)(C1)C(F)C2=O 67410,C(C(N=c1[nH]c(=NCC2CCCSC2)[nH]c2c1CSC2)c1ccnn1C)OC 67411,c1(C(=O)NC2CCN(C(c3n(CC)nnc3C)=O)C2)cc(C)cc(Br)c1O 67412,c1(C(N2CC(CN(C(C(CCC)C)=O)C)OCC2)=O)cnc(O)c2ccccc12 67413,N1(C(C(CCCC)CC)C(=O)NCCCC2CC2)CCC2(CC1)CC(=O)CCO2 67414,c1(CC)c(C(N2CCC2C(=O)O)=O)nnn1-c1cccc(C(C)C)c1 67415,c1(C2(C(=O)NCC(CC=C)NC(c3c(C#C)c[nH]n3)=O)CC2)cccc(Cl)c1F 67416,C1(C)(C(N(C)CC)=O)CC(NC(=O)CCOC(C)=O)C1.C1C(C)(C)O1 67417,c1(CC(N2CC(C)C(NC(c3nc(=O)n(C)[nH]3)=O)C2)=O)ccc2sccc2c1 67418,N1(C(CSCC=C)=O)CC2=C(C1)CN(C(c1cc(C)sc1Br)=O)C2 67419,CC(CCO)C(=O)N1CCCCC1Cc1cn(-c2cccc(F)n2)nn1 67420,C1(CC(=O)NCC2C(C(=O)NC(C=C)(C)C)C2)CCCCO1 67421,N1(C(C=C2CCN(C(c3cc(OC)ncc3)=O)CC2)=O)CC2CCCCC2C1 67422,C1(C(=O)NC2(CC(=O)NC3CCCC(C(C)C)C3)CC2)(OC)CCCCC1 67423,c1(C(C(N2C(C(=O)OCC)CCC2)=O)NCc2cc(C)c(Br)s2)ccc(O)cc1 67424,N1(C(CSCCOC)=O)CC2CCN(C(c3ccc(C4CC4)nc3C)=O)CC12 67425,O=C(C1=NOC2(CCC2)C1)N1CC(C2CC2C(=O)NCC23CCC(CC2O)C3)C1 67426,c1(C(N2CCC(NC(=O)Cn3cnc([N+](=O)[O-])c3)C2)=O)ccc2nc(S)[nH]c2c1 67427,C(c1cncc2ccccc12)=CC(=O)NC(C1N(C(CC(C)C)=O)CCC1)(C)C 67428,C1(C2CCN(C(CCC=C)=O)CC2)CC(N=c2[nH]c3ccc(N)cc3s2)CCO1 67429,C12(C(=O)NC(C(=O)NCC(C)(C)F)CC3CCOCC3)CCC(CC1)C2 67430,CCS(=O)c1ccccc1C(=O)NCC1CC1NC(c1nccc2ccsc12)=O 67431,c1(C(N2CCC(CNC(C(c3cccc(Cl)c3)CC)=O)C2)=O)ccc(F)c(N)c1 67432,c1(CC(N2CCCC(NC(C(C)OCC)=O)C2)=O)ccc2nsnc2c1 67433,Cc1ccc(CC(=O)NCC2CCN(C(=O)CN3CCCCC3)CC2)c(F)c1F 67434,C=CCC(C)C(=O)N(CCCCNC(C1(COC)CCCOC1)=O)C 67435,CCC(O)C(C)(C)C(=O)NCC1(O)CC(C(=O)N(CCC(F)(F)F)C)C1 67436,C(=O)(CC(C)(C)C(F)F)NCC1N(C(c2c(Cl)cn(CCC)n2)=O)CCN(C)C1 67437,Cc1c(C(=O)NCC2CN(C(=O)C=CC3CC3)CC2C)noc1-c1ccccc1 67438,C1(CNC(c2c(C)cco2)=O)CC2CCC(C1)N2C(=O)C(C)Oc1ccccc1 67439,c1(C(=O)NCC23CC(NC(C(C)OCC4CC4)=O)(C2)C3)ccc2nccn2c1 67440,C1(C(=O)NC(C#C)C2CC2)CCCN1NC(=O)C1CN(C(=O)CC)C1 67441,c1(CC(=O)NC(C)(C)CCNC(C23CCCC2C3(F)F)=O)c[nH]c2cnccc12 67442,N1(C(c2c(NC)cccc2)=O)CCC2C(CCCN2C(C2(C)CCCC2)=O)C1 67443,CC1(F)CCC(C(=O)NC2C3CN(C(=O)CC4CC=CCC4)CC23)CC1 67444,C1(C(=O)NCCN(CCC)C(c2cc(C)ccc2OC)=O)CCC2C1C2(F)F 67445,CC1CN(C(C2OCCCC2(C)C)=O)C(C)CN1C(C1CN2CCC1CC2)=O 67446,N1(C(C(=O)NC(=O)NCC(C)C)C)CCC(C)(NC(c2sccc2Cl)=O)C1 67447,c1(N(C(C2CCC(C(C)C)CC2)C(=O)NC(CC)C)C)ccc(F)c(Cl)c1 67448,C1(NC(C(CN(C)C)O)=O)CN(C(c2cc(F)c[nH]2)=O)CCC1C(F)(F)F 67449,C(=O)(C(C)(C)NC(C)=O)NC1CC(CNC(C2(CSC)CCC2)=O)C1 67450,N1(CCc2cn(-c3n(C)nnc3)nn2)CCN(C(C2CC(=O)N2)=O)CC1 67451,C1(CC)CN(C(=O)CSc2nncn2C)CCC1NC(=O)Cc1cc(Cl)cs1 67452,c1(CNc2nc(-c3ccc(OCCC)nc3)sc2)ccc2[nH]c(C)cc2c1 67453,N1(C(CNC(CC)=O)=O)CCC(C(C)C)CC1CNC(=O)C=CBr 67454,C(=O)(CCCCC(C)(C)C)NC(C(=O)N(C)Cc1c(C)ccs1)Cc1ccco1 67455,C=CCC(CC)C(=O)NCC(c1ccccc1)CNC(C1(O)CC(C)(C)C1)=O 67456,C1(CC(C)NC(C23CSC(C2)C3)=O)CCN(C(=O)CN2CC(=O)NC2=O)CC1 67457,CN1CCC2CCN(C(=O)C(O)CCCNC(c3ccc(F)c(F)c3)=O)C2C1 67458,N1(C(Cn2cc(CCCC=C)nn2)=O)CCC(O)C1C(C)(C)C 67459,C(C)(C)(CC(C)(C)O)NC1C(n2cc(CS(CC)(=O)=O)nn2)CCC1 67460,C=CCCCCC(=O)N1CCC(C(C)C(=O)NC(CC)C(C)(F)F)C1 67461,C(C(=O)N1CC(F)(F)C1CC(=O)O)(C(C)(C)C)n1cc(-c2c(C)nccc2)nn1 67462,Cc1c(Br)noc1C(=O)NC(C)CCNC(=O)CC1C=CCC1 67463,N1(C(C2=NNC(=O)C2)=O)CC(NC(=O)CC2CCC(=O)NC2)CC(F)(F)C1 67464,O=C1CNC(=O)C(CC(=O)NCCN2CCN(C(=O)CNC=O)CC2)N1 67465,C1(C)(C(N2CC(SC)C(n3cc(CC4CCOC4)nn3)C2)=O)CCCCNC1=O 67466,C(CC(C)C)(C(=O)NC1(CF)CCN(C(c2cscc2C(F)(F)F)=O)C1)OC 67467,C1(OC)CN2CC1N2C.C1(C(=O)NC=O)CCN(C2COC2)CC1.OC 67468,N1(C(C2CC(F)CN2C(=O)Cc2ccc(Cl)c(F)c2)=O)CCCC2CCCCC12 67469,c1(-c2nc(C(=O)Nc3c(C(=O)OC)ncs3)sc2)ccc2nc(Br)sc2c1 67470,C(=O)(C(F)C(C)(F)F)NCc1ccc(C(N(CC)CC2CCOC2)=O)s1 67471,C1(NC(=O)OC(C)(C)C)C2CC3C1C3C2NC1C(F)(F)C12CCC2 67472,C1(N(C(c2cc(CCC)[nH]n2)=O)C)CCCC(NC(=O)CN2CCCCCC2)C1 67473,C12(CC(N3CCC4(CCC4)C3)=O)CCC1CN(C(c1cccc(CO)n1)=O)C2 67474,C1(C)(C(=O)NCC2(O)CC(C)(C)C2)CCCN(C(=O)Cn2cnc(C#N)n2)C1 67475,c1(C(=O)NCC2N(C(C(c3ccncc3)C)=O)CC2)c(F)cccc1Cl 67476,C=C(Cl)CCC(=O)NCC1(C)CN(C2CCN(C(C3CCCC3)=O)CC2)C1=O 67477,C(=O)(CN=c1ccc(Cl)n[nH]1)N1CC(CNC(c2ccc(C)o2)=O)CC12CCC2 67478,CCC(C)C(C(=O)NCCc1cnc(C)o1)N(C(=O)CCCC1CCC1)C 67479,C#CCC(C)(C(=O)NCCC1CC(=O)N(C)C1)NC(c1cc(C)sn1)=O 67480,c1(-c2c(C)ccc(CO)c2)cc(C(=O)N)cc2c[nH]nc12.N1(CCO)CC2CC2C1C#N 67481,C1(C2CCN(C(C3CCCO3)=O)C2)(NC(c2cccc(C(C)C)n2)=O)CC1 67482,C1(CNC(CCCC=C)=O)CN(C(=O)CN2CCC(=O)NC2=O)CC1(C)C 67483,c1(C(N2CCCC(NC(c3cn(CC(F)(F)F)nn3)=O)C2)=O)c(F)cncc1Cl 67484,C1(C(=O)NC2CCC(N(C)C(C3CC34CCCC4)=O)CC2)CC2CSCC(C1)C2 67485,N(C(=NCCc1cccs1)NCCN1CCCCC1)CCOC.c1(C)nc(C)c(C)s1 67486,C#CC1(C(N2CC(C(C)(C)C)C2)=O)CCN(C(c2nn(C)cc2C)=O)C1 67487,Cc1c(Br)noc1C(N1CCC(C)C1CNC(=O)CN1CC2CC2C1)=O 67488,C(=O)(C1=CC2CCC(C1)C2)N1CC(C(=O)NC2COCC2O)C(F)(F)C1 67489,c1(C(=O)NCC(CNC(c2cc(CCC)nn2C)=O)(C)C)cc2occc2[nH]1 67490,N1(C(C(C)CC(N)=O)=O)CCCCCC(Nc2ncnc(C(C)(C)C)n2)C1 67491,N1(C(CC(=C)C)=O)CCCC(CCCCNC(C2(Cl)CC2(F)F)=O)C1 67492,c12c(cccc1F)NC2=O.C1(CCC(=O)OC)CCCN1S(=O)(=O)C1CC1 67493,c1(NC(C(N2CCN(C(c3cc(C)c(C)o3)=O)CC2)C)=O)ccn2nccc2n1 67494,CC(=O)C(C)CC(C)C(=O)N(C1CC(NC(=O)OC(C)(C)C)C1)C 67495,c1(NC(CCCNC(C2(OCC)CCCCC2)=O)C)ncc(Cl)c(C)c1C#N 67496,c1(N2CCCC(CNC(C)=O)C2)ccc(S(=O)(=O)N(CCCCO)C)c(Cl)c1 67497,CC(C)(C)C#CC(=O)NCCCC1CCCCN1C(=O)CC1CCC(=O)O1 67498,N1(C(C(CCC)N(C)C)=O)CC2CCCC1(CNC(C1CC13CC3)=O)C2 67499,N1(C(c2ccnc(Cl)c2O)=O)CC2(C1)CN(C(C13CC(O)C1C3)=O)CC2CO 67500,Nc1c(C(=O)NC2CC2NC(C2CCC(NS(N)(=O)=O)CC2)=O)cccc1[N+](=O)[O-] 67501,c1(CC(=O)N(CC(CNC(C2CCN(CC)CC2)=O)C)C)c(C)nn(CC)c1C 67502,C=C(C)C(O)CC(=O)NCCC1CN(C(=O)CCCc2nc(CC)no2)CCO1 67503,c1(C(=O)NCC2CC2NC(c2cc(F)c(F)cc2Cl)=O)cc2n(n1)CCNC2=O 67504,c1(C(N2CCN(C(CCC(C)OC)=O)C(CCO)C2)=O)nc2ncccn2n1 67505,c1(NC(C2C3(CN(C(c4cncc(C)n4)=O)C3)C2)=O)cc(C(F)(F)F)ccc1I 67506,C(=O)(CC(CC)C(F)F)NC(CCC#C)C(=O)NC(C)Cc1ncn(C)n1 67507,C(=O)(C(F)CCC(C)(C)C)NCC1(OC)CCN(C(C(CC)F)=O)C1 67508,C#CCC(CC(F)F)C(=O)NC(CCC)CC(=O)NC1(C(F)(F)F)CC1 67509,N1(C(CC2(OC)CCC2)=O)C(C(=O)Nc2sncc2C#N)CC2CC12 67510,CN(C(=NCC1C=CCCCC1)NC1CCC1)Cc1ncnn1C 67511,c1(CC(=O)NC2CC(NC(c3ccsc3)=O)CC2O)n[nH]c2ccccc12 67512,c1(C(=O)NC2CCC23CN(C(=O)CCC2CCCO2)C3)[nH]nc2ncccc12 67513,c1(CC(=O)NCCC(C)NC(c2c(F)ccc(CC)c2)=O)cnn2c1CCCC2 67514,C(=O)(C(C)(CC#C)NC(=O)C(O)C=CC)N(C(CC#C)C)C 67515,CC1=C(C(=O)NCCCCCNC(C2(C)CNC(=O)N2)=O)SCCO1 67516,c1nc(C)c(C)s1.n1(CCC)nnnc1C1C2CC(C2)N1.CCOCC 67517,N(C(=NCCOCc1ccc(N(C)C)cc1)Nc1ccc(Cl)cc1)C(CSC)C 67518,Cc1cccc(C)c1C(=O)NC(C)CC1CCN(C(C2CCC2(F)F)=O)CC1 67519,Cc1ccccc1-n1cc(C(=O)NCC2CC2NC(C2CC(C)(C)CO2)=O)nn1 67520,c1(C(N2C(CCCC)CN(C(C3CC34CC4)=O)CC2)=O)cnc2c(C)nsc2c1 67521,Cc1cccc(N2CCC(NC(=O)Cn3cc(-c4ccc(C)cn4)nn3)C2=O)c1 67522,C(F)(c1ccccc1)=CC(=O)NCCC(C)(C)NC(C1CCC(F)(F)C1)=O 67523,c1(C(C(N2C(CN(C(c3c(CC)ocn3)=O)C)CCC2)=O)C)ccncc1C 67524,N1(C(CC(CC)O)=O)CC2CC(NC(=O)C3=CCCCCC3)CC1C2 67525,CC(C)C(F)C(=O)NCCN(C(C1CC(=C(F)F)C1)=O)C(C)C 67526,C(CN=c1cc[nH]c(-c2nccs2)n1)C1CCC(NC(CCCCCC#C)=O)C1 67527,c1(C(=O)NC(C)CCNC(=O)C(C(C)O)NC(N)=O)cnc(N)c(Cl)c1 67528,C=CC(CCC)CC(=O)NCCN1CCC(NC(c2sccc2OC)=O)CC1 67529,C(=O)(C1=NOCC1)N(CC(=O)NC(c1nc[nH]n1)CC)CCOC 67530,c1(CCC(=O)NC(C2(CCC(=O)OC)CC2)=O)cccc(C#N)c1 67531,CCC(C#N)C(=O)Nc1cccc(NC(C)=O)c1.C12CN(C1)C2=O 67532,C12(C(=O)OCC)CCCC(CN3CCN(C4CCC4)CC3)(C1)OC2 67533,C(CCS(C)(=O)=O)(C(=O)NCCCN(C(c1ncccc1O)=O)C1CC1)OC 67534,C12(NC(CNC(=O)OC)=O)CCCC1CN(C(=O)C(C)CN1CCOCC1)C2 67535,Cc1ccccc1CCNC(C1CCCN(C(C(C)Cc2cncnc2)=O)C1)=O 67536,C1(OC)(CNC(C2CC3CCC23)=O)CCN(C(c2cc(O)cc(Cl)c2)=O)CC1 67537,Cc1ccc(C)c(C(=O)NCC2(C)CCCN(C(C3CCC(=O)N(C)C3)=O)C2)n1 67538,C1(CNC(C(CC=C)OC)=O)COC(C)(C)CN1C(c1ncc(F)cc1F)=O 67539,Cc1cc(C(=O)NCC(O)CNC(=O)C=CC2CC2)cc(O)n1 67540,c1(C(=O)NC2(C)CC(NC(C=C3CCC(C)CC3)=O)C2)cccc2c1CCN2 67541,n1(CC(N2CCC(N(C(CCNC(C)=O)=O)C)C2)=O)nc(C)oc1=O 67542,c1(C(N2CC(C3(NC(CCN(C)CC)=O)CC3)C2)=O)cc(C)c(OC)c(Cl)c1 67543,C(=O)(CCS(=O)(=O)Cc1ccccn1)N(CCCCNC(=O)C#CC1CCC1)C 67544,Cc1cc(CC(=O)NC(C2CCOC2)CNC(C2CC(C#N)C2)=O)on1 67545,N1(C(C(F)=CCC)=O)CCC(CO)(NC(=O)COC2CCCC2)C1 67546,C1(N(C)C(C2CCCCN2C(=O)C(C)(C)C)=O)COC(C)(C)OC1 67547,CCCCS(=O)(=O)CC(=O)NCCCCC1CCN(C(=O)C(O)C(C)C)CC1 67548,C1(C(N(CC(C)N(C(Cc2scc(C)c2)=O)C)C)=O)C(C)(C)C1(F)F 67549,C(=O)(CC(C(C)OC)NC(C1CC(=O)CS1)=O)N1CCC(C#C)C1 67550,c1(N2C(CNC(c3ccc(F)cc3)=O)CC(F)C2)nc2cc(F)cc(F)c2o1 67551,N1(C(CCSc2ccc(C)cc2)=O)CC2CCC1CN2C(=O)C(C(C)O)N(C)C 67552,CCCC(O)C(=O)NCC(F)CNC(c1sc(COC)nc1C)=O 67553,n1(CC#C)c(C)cc(C(N2CC(CCNC(c3cc(C(C)C)no3)=O)C2)=O)c1C 67554,C1(NC(CS(N)(=O)=O)=O)CN(C(c2ccc(C3CCC3)cc2)=O)C2CCCCC12 67555,c1(C2C(NC(C3(c4ccccc4)CC3)=O)C2)ccc(Br)cc1F 67556,C(c1ccc(C(C(=O)NCC2CC2)N(C)Cc2nc[nH]n2)cc1)=CC(=O)OC 67557,c1(CC(C(N2CCC(NC(C3CC(C)(C)C3)=O)C2)=O)O)ccncc1Br 67558,CCC(CC)C(C)C(=O)N(CCC(=O)NCc1csc(C)n1)CCCO 67559,N1(C(C(C)SC)=O)CCCC(CCNC(c2c[nH]nc2-c2ccccn2)=O)C1 67560,C(CS(=O)(=O)CC(=O)N1CC(NC(c2cc(C)sn2)=O)CC12CCC2)OC 67561,C1(N(C(Cc2c(C)non2)=O)C)CC2CC1N(C(=O)Cn1nccc1C)C2 67562,c1(C(C(=O)NCC(C)C)N(C2CCSCC2)C)nnc2n1CCC2 67563,CC1CCCC(C)N1C(=O)C(N1CCC(CN(C)C(c2cc(Br)n[nH]2)=O)CC1)=O 67564,N1(C(C(=O)Nc2ccc(N(C)C)cc2C(F)(F)F)=O)CCCC12CCOCC2 67565,c1(CCC(N2CC(O)(C(C)NC(C=CC=CC)=O)C2)=O)ccnc(C)n1 67566,c1(OC(C)(C)C)cccc(Cl)c1NC(=O)C(CC(C)C)OC(=O)Nc1ccccc1 67567,C1(CNC(c2csc(C)c2C2CC2)=O)C(C)CCCN1C(c1cnns1)=O 67568,c1(CC(=O)NCC2N(C(C(CC(=C)C)C)=O)CCOC2)csc2nc(C)cn12 67569,c1(N2CCCC(CCC)C2)ccncc1S(=O)(=O)NCc1nccn1CCC 67570,CC(C(C)(C)NC(=O)CCCn1cncn1)NC(=O)COCCc1ccccc1 67571,c12nnc(n1CC1(C)CC1)CN2C.c1(CC2CCCC2)ncn(C)n1 67572,C(=O)(C1=CCCCC1P(C)(C)=O)NCC(CNC(C(C)(C)C1CCC1)=O)CO 67573,c1(C(=O)NC2C(NC(C3(CC)COC3)=O)C2)ccc2ccn(C)c2c1 67574,N1(C(c2nc(OCC)oc2)=O)CC(NC(=O)CC2(C)CCCC2)C(C)(C)C1 67575,C1(NC(c2nc(C)oc2)=O)C2CC1N(C(c1c[nH]nc1OCC(F)(F)F)=O)C2 67576,Cn1nnc2c1CCN(C(=O)CCCCCNC(=O)C(C)(F)C(C)(C)F)C2 67577,Cc1c(C(=O)NC2CCN(c3ccnc(C4CC4)n3)CC2)ccc(F)c1F 67578,C1(C(=O)OC)C(C)CCN1C(C1CC(NC(=O)C(C)(C)N(C)C)CCO1)=O 67579,C1(C(N2CC(O)(CNC(CC3(COC)CC3)=O)C2)=O)CCc2cnn(C)c2C1 67580,c1(OCC(=O)NCC(C(C)C)NC(=O)C(O)c2cnc[nH]2)cccc(Br)c1 67581,N1(C(C(C=CC)O)=O)CCC(NC(c2cccc(Br)c2)=O)C1(C)C 67582,N1(C(c2nc(C)oc2)=O)CC(NC(C2COC3COCC3O2)=O)CC12CCCC2 67583,c1(C(=O)NC2CC(CNC(C3CC(CCC)OCC3)=O)C2)ccc([N+](=O)[O-])s1 67584,N1(C(C(c2cccc(Cl)c2)(C)C)=O)CC2CCN(C(C3CCCS3)=O)CCC2C1 67585,C1(NC(c2c(OC)n[nH]c2)=O)CCN(C(=O)CN2CCCC2=O)CC1O 67586,C1(C(=O)NCCc2onc(C)n2)CC(C)CN1C(=O)CN1CCCC1C 67587,C1(C(N(CCC)CCNC(=O)CSCc2cscn2)=O)CC2CCCC(C1)C2 67588,c1(-n2ccc(C(=O)NC3C(NC(=O)C=Cc4cscn4)C3)n2)ccccc1Cl 67589,c1(C(=O)NC(CC)CN(C(=O)CN(CC)CC)C)c(C)noc1C1CC1 67590,C(CCCCCCC)N(C(C(Cc1cc[nH]n1)NC(C1CCC(=C)CC1)=O)=O)C 67591,c1(CNC2CC(NC(c3ccc(C)cc3C)=O)C23CCC3)cc(C)cc(C)c1N 67592,C#CCC(CC(=O)NC1CCC(NC(=O)C=CC(C)(C)C)C1)c1ccccc1 67593,C(=O)(CCCC(C)(C)C)N1C(CCNC(c2cnn(CC)c2C)=O)COCC1 67594,c1(C(N(CCNC(c2c(O)cc(C)nn2)=O)C2CC2)=O)c(C)nc2ccccn12 67595,C=CCC(C)(C)CC(=O)NCCC1CC(F)(F)CN1C(=O)CCOC1COC1 67596,CC1CCCCCC1NC(c1coc(CNC(C2CC2[N+](=O)[O-])=O)n1)=O 67597,c1(NC(=O)C(N2CCCCC(CO)C2)=O)cc(N2CCCC2)cc(F)c1 67598,N1(C(CC(C)(C)OC)=O)CC(C)N(C(C2(C)CC3CCC2O3)=O)C(C)C1 67599,C1(C)(CNC(Cc2cn(C)nn2)=O)CCC(NC(=O)COCc2ccnn2C)C1 67600,c1(CCC(=O)OC)ccc(Cl)c(NC(=O)NCc2oc(C(C)C)nc2C)c1 67601,c1(OC)cc(OC)cc(C(O)CNCc2cnc(OC)cc2C)c1 67602,C1(NC(C(c2cccc(Cl)c2)C)=O)CN(C(c2cc(F)n[nH]2)=O)CCC1O 67603,CC1(NC(=O)NCC2(CSc3ccccc3)CC23CCC3)CN(C2CC2)C1=O 67604,c1(CNC(C2(C)CCCN2C(C2CCCC2)=O)=O)cnc(O)nc1O 67605,C1(C)(C(=O)NCCCOCCNC(c2c(C)cccn2)=O)CC2CCC1O2 67606,c1(C(=O)NCC(CO)NC(=O)Cc2csc(Cl)n2)nccc2c1NCCC2 67607,CCC(CC)(CCNC(=O)OC(C)(C)C)NCC1CCCOC1CC(C)C 67608,CCC(C)CCCCC(=O)N1CCC(NC(C2CCCC(C)(C)C2)=O)C(C)(C)C1 67609,N1(C(C(C(C)C)c2cccnc2)=O)CCOCC(NC(c2cccnc2)=O)C1 67610,C1(C(N2CC(c3ccccc3)(NC(CC(C)OC)=O)C2)=O)CCCCC1(C)C 67611,c1(N2CCC(CC)OCC2)nc(N2CCSC(c3cccs3)C2)c2c(n1)CCS2 67612,Cc1nc(NC2CCc3n[nH]cc32)cc(C#N)n1 67613,c1(C(N2C(C(C)(C)NC(=O)CCC3CCC3)CCC2)=O)ccc2nc[nH]c2c1F 67614,C1(N(C(CSCCCC)=O)C)CCN(C(=O)CCCc2cccs2)C1 67615,C(C(F)(F)C(C)(C)O)NC(C1(CNC(C(CN(C)C)O)=O)CC(C)(C)C1)=O 67616,CC(O)(C(=O)NCC1(C(N2CCC(n3cnnn3)C2)=O)CC1)C(F)(F)F 67617,C(=O)(CS(=O)C(F)(F)F)N(C)CCN(C)C(C1CCN1C1CCCC1)=O 67618,CCCCCC(F)C(=O)NC(C)(C)CCNC(c1cnn(CC)c1C)=O 67619,CN1CCCc2cc(C(=O)Nc3nnc(CF)s3)ccc21 67620,N1(C(CC)=O)C2CCCC1CN(C(c1c([N+](=O)[O-])c(C(F)(F)F)nn1C)=O)CC2 67621,CC1(C)CC(C(N2CC3(CCC3O)C2)=O)CN1C(c1ccco1)=O 67622,CCC(O)C(C)(C)C(=O)NCC(CC(=O)N(CC(C)(CC)OC)C)OC 67623,n1(-c2n(Cc3c(O)noc3)nnn2)ncc2cc(Br)ccc12 67624,c1(C(=O)NCC2(O)CN(C(C(C(C)O)C)=O)C2)cn2cc(Cl)cnc2n1 67625,C1(CCOC)(NC(=O)CNC(C)=O)CCN(C(c2[nH]ccc(=O)c2C)=O)CC1 67626,C1(C(=O)NCCCC(C)NC(=O)CCC#N)(CO)CCCCO1 67627,Cc1ccccc1CC(C)C(N1CCC(F)(CNC(=O)CC2CC3(CC3)C2)C1)=O 67628,CC#CCC(C(=O)Nc1cnccc1OC)NC(=O)C(CC1CCC1)OC 67629,O=C(CC=C(Cl)Cl)NC1CCCC1CNC(=O)C=Cc1cc[nH]c1 67630,c1(C(N(C2CN(C(=O)CCCC#N)CC23CC3)C)=O)cc2ccsc2n1C 67631,N1(C(C(c2cncnc2)C)=O)CCC(NC(=O)C=Cc2ccco2)C12CC2 67632,N1(C(CC)=O)CCC(C)C1C(=O)N(C)Cc1ncc(Br)cn1 67633,C1(C)(C(N(CCC)CCNC(=O)CC2CCCC2)=O)CCCC1O 67634,S(=O)(=O)(c1ccc(NCC(c2ccccc2F)OC)cc1Br)NCC=C 67635,c1(OC(CNC(C(=O)NCc2cnn(CC)n2)=O)(F)F)cccc(Cl)c1 67636,C(CNC(c1c(C)noc1CC)=O)(C(C)C(C)C)NC(CCCC=C)=O 67637,C#CC1(C(=O)NCC(c2ccnn2C)O)CCN(C(c2csc(C)n2)=O)C1 67638,C1(C(=O)NC2C(CC(=O)NC3C(CN(C)C)CCC3)C(O)C2)CC2CCCC2C1 67639,Cc1ccc(C#CC(=O)NCC2CCOCO2)cc1 67640,C1(NC(c2cncc(OC)c2)=O)CN(C(C2CCSC2)=O)C2CCCC12 67641,C(c1ccncc1)=C(C)C(=O)NC1(CO)CN(C(C2(Cl)CC2(F)F)=O)C1 67642,O=C(C1=NOC2(CCOC2)C1)NC12CCC1CN(C(=O)C=CC1CCC1)C2 67643,c1(OCC(=O)NCC2CN(C(C=CC(=O)OC)=O)C(C)C2)ccc(Br)c(F)c1F 67644,c1(CNC(CSCCC)=O)cnn2c1CN(C(c1[nH]nnc1C)=O)CC2 67645,N1(CCCCNC(c2cnc(C)[nH]2)=O)CCCN(C(c2c(Cl)n[nH]c2C)=O)CC1 67646,c1(C(C)(C)C)nc(=NC2CC(NC(C3CC3c3ccccc3)=O)C2)s[nH]1 67647,Cc1c(Cl)sc(Cl)c1C(=O)NCC(Cc1ccccc1F)CO 67648,C1(CC(=O)N(C2CCN(C(c3cc(C(C)=O)c[nH]3)=O)C2)CC)CC2CCC1CC2 67649,N1(C(c2cc(OC)n[nH]2)=O)CCCC(CNC(=O)C(O)Cc2cnc[nH]2)C1 67650,C1(CC=C)(C(=O)NC2(CCO)CCC2)CCN(C(=O)CN2CCNC(=O)C2)C1 67651,c1(NCC=CCNC(Cc2c(C)ncnc2C)=O)cc(=O)n(C(C)C)c(O)n1 67652,N1(C(CN(CC)CC)=O)CC(CNC(=O)CCc2ccc(SC)cc2)C2(CC2)C1 67653,N1(C(CC(C)CN(C)C)=O)C2CC1CN(C(C1CC1C#N)=O)C2 67654,N1(C(C=CCN(C)CC)=O)CCN(C(c2cc(C3CCCC3)[nH]n2)=O)C2(CC2)C1 67655,C1(NC(C2CC(CC)C2)=O)COCCN(C(c2c(N)cccc2Cl)=O)C1 67656,CC1CCOC(C(=O)NCCN(C2CCCCC2)C(c2cc(=O)cc[nH]2)=O)C1 67657,C1(NC(c2ccnc(N3CCCC3)n2)=O)CCCN(C(c2ccoc2)=O)C1 67658,C1(C(=O)NCC2CCC(C)C2)(OC)CCN(C(=O)C=NOC)C1 67659,N1(C(CC=CC)=O)CC(CNC(c2cc(CO)[nH]n2)=O)CC1(C)C 67660,C(=O)(CCCCC1CC1)NC(c1ccccc1)CNC(c1ncc(CC)s1)=O 67661,N1(C(C2CCN(C(=O)OC)C2)=O)CC(=O)NC(C2CC2)C1 67662,N1(C(C2C(C(C)(C)C)CCCC2)=O)CC2CCCC(C1)N2C(C1CCCS1)=O 67663,N1(c2cc(C(=O)OCC)ncn2)CCCN(C(=O)CC(C)c2ccccc2)CC1 67664,c1(-n2c(-c3scc(-c4cn(CC(=O)OC)nc4)c3)ncc2)c(C)cccc1Cl 67665,c1(C(N(CC(O)CN(C(=O)C(F)C(F)(F)F)C)C)=O)ccc(C#N)cc1 67666,C1(NC(=O)C=CC=C(Cl)Cl)CC2(CCCCN2C(=O)CCCC2CC2)C1 67667,N1(C(=O)CSCc2ncc[nH]2)CCC2(CCCN(C(=O)CC3CCOC3=O)C2)C1 67668,CCC(C)C(=O)NCC(CNC(=O)C(C)(C)NC(=O)OC(C)(C)C)OC 67669,C(=O)(C(C(C)(C)O)NC(=O)CC1COCC(C)O1)N(CCC)C 67670,N1(C(C2CN(C(C3CC(F)(F)C3)=O)C2)=O)CCOCC1C.c1(C)ccccc1 67671,N1(CC)C(=O)CCC1CC(=O)N(CC(O)CNC(=O)C(Cl)=CCl)C 67672,c1ccc2c(c1)nc(N1CCC(n3cc(C4CCNC4)nn3)CC1)c1cncn21 67673,C1(CNC(C(CC=CC)C)=O)CN(C(=O)COC2(C)CCCC2)CC1(C)C 67674,N1(C(CSCCCC)=O)CCCCC(CCC(N2CCC(F)(C#N)C2)=O)C1 67675,c1(C(=O)NC2CN(C(c3c(C)snc3)=O)CC2O)cn(CCO)c(=O)nc1O 67676,c1(C(N(C)C)=O)cccc(C(=O)N(N2CCOC(CS(C)(=O)=O)C2)C)n1 67677,S(=O)(=O)(c1cc(F)c(F)cc1F)NC1C(C(=O)Nc2ccc(C)cc2I)CCC1 67678,C1(NC(Cc2n(C(C)C)cnn2)=O)CCC(C)N(C(=O)CC2(C)OCCO2)C1 67679,N1(C(c2cc(CC)[nH]n2)=O)CCC(NC(c2ccc(C(C)C)s2)=O)C(C(C)C)C1 67680,CC1=C(C(=O)NC2CCN(C(=O)C3CC3)C(C)C2)C(C)n2nnnc2N1C 67681,CCCCCCC(C)NC(=O)C=CC(C)NC(c1coc(C2CC2)n1)=O 67682,N1(C(CCN(C)CC)=O)CCCC(CCNC(c2n[nH]c3c2CCC3)=O)CC1 67683,c1(C(N2CC3(CCCN(C(C4C(CC)C4)=O)C3)C2)=O)ccc2c(Cl)nccc2c1 67684,C(=O)(CCC(F)(F)C(F)F)NC1CN(C(c2ccn(CCC)n2)=O)CC(O)C1 67685,c1(C(N(CCCCNC(C(C)OCCCC)=O)C)=O)ccc(C)nc1 67686,c1(OC)ccc(C(N2CC(O)(C3CCCN3C(=O)CC(C)OC)C2)=O)cn1 67687,C12(C(=O)NCC(C)CNC(=O)Cc3ccsn3)CCCCC(F)(C1)C2 67688,c1(C(N2CC(C)C(CNC(=O)CCn3cnnn3)C2)=O)nn2cccnc2c1Cl 67689,c1(CN2CC(C)C(F)(C(=O)O)C2)cc2ccccc2cc1O 67690,C12(C(=O)NCC3CN(C(c4ccc(F)cn4)=O)CC3O)CCC(F)(CC1)CC2 67691,C(=O)(C1CC(=O)c2ccccc21)NC(C)CNC(=O)COC1(C)CCCC1 67692,C1(NC(=O)Cn2ccnn2)C=CC(CNC(c2cc(Br)c[nH]2)=O)C1 67693,c1(OC)ccc(C(N2CC(CCNC(C3(O)CC3)=O)OC(C)C2)=O)c(F)c1 67694,C1(NC(CC(COC)C)=O)CCC2CN(c3cc4nnc(C)n4cn3)CCC2C1 67695,c1(OCC)cc(C(C(=O)Nc2ccccc2Cl)N(C2CC(C)C2)C)ccn1 67696,C(CC(=O)Nc1cccc(Cl)c1O)(C(C)(C)C)NC(c1cnc(C)o1)=O 67697,CC(C)CC(C(=O)NCCC1CC(NC(C2CCCC(C)(C)CC2)=O)C1)C(N)=O 67698,CCC(O)(C(=O)NCCN(C(=O)CC(C)(O)c1ccccc1)C)c1ccccc1 67699,C(CC(=O)N(CC(O)C1CC1)C)N(CC(C)C)C(C)=O 67700,Cc1c(C(N2CCCC(CO)C2)C(=O)NC2CCCCC2)cccc1Cl 67701,CN(S(N)(=O)=O)CC(=O)NC(CNC(=O)Cc1ccsn1)CO 67702,c1(C(N2CC(C)C(CNC(C3(O)CC3)=O)CC2)=O)cccc2ncoc12 67703,N1(C(CCCCC=CC)=O)CCC(NC(=O)COc2cccnc2)C(CO)CC1 67704,N1(C(c2ccc(C(C)C)cn2)=O)CC(CNC(=O)CP(C)(C)=O)C2(CCC2)C1 67705,c1(CC(=O)NCC2C(NC(c3c(CC)csc3)=O)CCC2)ccc(OC)c(Cl)c1 67706,C1(C(=O)NC(c2nc[nH]n2)CC)CCCN1C(=O)CC1CCSC1 67707,N1(C(C2(C)CCC(=O)N2)=O)CCC2CC(NC(c3ccc(F)cc3)=O)CCC2C1 67708,C1(NC(C2CCC(F)(F)CC2)=O)CN(C(C2CC2(Cl)Cl)=O)C2(CCOCC2)C1 67709,c1(C(N(C2CN(C(=O)Cc3cccc(O)c3)C2)C)=O)ccnn(C)c1=O 67710,C1(N(C(C=CC(=O)OCC)=O)C)CCCCC1N(C)C(C1CC1F)=O 67711,c1(SC(C)C(=O)NCC(C)(O)CNC(c2ccn(C)c2)=O)ccccn1 67712,n1(CC(=O)NCC(N2CCN(C(C3CCC3Br)=O)CC2)C)ncc2ccccc12 67713,N1(C(C2CN(C(c3cc(C(C)C)[nH]n3)=O)CC(F)C2)=O)Cc2ccccc2C1 67714,C1(C(=O)NC2CCCN(C(c3c(CC)oc(C)c3)=O)CC2)CC2(CCCC2)CO1 67715,Nc1cc(Cl)cc(F)c1C(N1CCCN(C(c2cccc(O)n2)=O)CC1)=O 67716,CC1CN(C(c2c(Cl)ccnc2O)=O)c2cnccc2NC1=O 67717,C1(CN(C)C(C2(C)CC2(F)F)=O)COCCN1C(=O)CN1CC(=O)NC1=O 67718,C(=O)(C(C)S(N)(=O)=O)NC1C(CNC(CC2C(C)CC2)=O)COC1 67719,N1(C(Cn2ccc(C)n2)=O)CCC12CCCN(C(c1n[nH]c(C)c1C)=O)C2 67720,c1(C(=O)NCCOC2CCN(C(CC(C)SC)=O)CC2)ccc(C)cc1[N+](=O)[O-] 67721,c1(NC(N2C(COC)C=CC2)=O)cc(CCCO)n(CCn2cnnc2)c1C 67722,CCC(C)CCCC(=O)N1CC2CCC(C1)N2C(c1cnsn1)=O 67723,c1(SCC)nc(C)c(C(CC)C(=O)Nc2csc(CC)n2)s1 67724,C(=O)(C(CS(=O)(=O)C(C)C)NC(=O)OC(C)(C)C)NC(CC=C)CCC 67725,C(C)(CC(=O)NC1CC(F)CN(C(=O)CNC=O)C1)(C(F)(F)F)N(C)C 67726,N1(C(c2occc2C2CC2)=O)CCN(CC(N2CC3CC(C2)O3)=O)CC1 67727,N#CC1(C(N2CCC(NC(C3CCCC(C(N)=O)C3)=O)C2)=O)CCCO1 67728,N1(C(CNC(=O)NC)=O)CCC(O)(C2(NC(=O)CC3CC=CC3)CC2)CC1 67729,CN1CCCCCC1C(=O)Nc1ccc(Oc2cccc(C#N)c2)cc1 67730,c1(NC(=O)CNC(CC2CCCC2)Cc2ccc(F)cc2)ccnc(C(=O)O)c1 67731,C#CC1(C(=O)NC2COCC(C)(C)C2)CCN(C(c2ccoc2CC)=O)C1 67732,C1(NC(C(C)(O)C2CC2)=O)CCOCC1C(N1CC(F)(F)C1C1CC1)=O 67733,C1(NC(C(C=C)O)=O)CCCC12CCN(C(=O)COCC(=O)OC(C)(C)C)CC2 67734,CC1CN(C(=O)C2=COCC2)CC1CNC(C1OCCC1c1cnn(C)c1)=O 67735,c1(C(N(CCCCNC(C2COCC(C)O2)=O)C)=O)ccnc(C(F)(F)F)c1F 67736,c1(C(=O)NCC(C)N(C)C(c2ccnc(Cn3cnnc3)c2)=O)nnn(C)c1N 67737,N1(CC(=O)NCCC(C)N(C(=O)C=Cc2cscn2)C)CCC(C(N)=O)CC1 67738,C12(CNC(C=CSC)=O)CCCC1CN(C(c1cc(C(N)=O)[nH]n1)=O)C2 67739,c1(OCC)cc(C(N2CCC(C)(NC(c3cnc(C)s3)=O)C2)=O)ccc1OC 67740,Cc1nccnc1C(c1ccc(C(=O)NNC(=O)NC(C)C)o1)N(C)C 67741,c1(CC(=O)NCCC(C)NC(=O)Cc2ccc(F)cc2)ccc(C#N)nc1 67742,C#Cc1cccc(CC(N2CC3CC(N(C)C(c4cc(C)no4)=O)C2C3)=O)c1 67743,C1(NC(C(C2CC2)OCC)=O)CCN(C(c2ncc(C)cc2OC)=O)CC1CC 67744,c1(C(c2nnnn2CC(F)F)NCC(=C)CC)c(N(C)C)ccnc1Br 67745,N1(c2cc(C)ncn2)CCC(NC(c2cccc(P(C)(C)=O)c2)=O)CC(C)(C)C1 67746,C(CCN=C(NCC1CCC1)N1CCSC(C(C)C)C1)NC(COC)=O 67747,C12(C(=O)NCC3C(NC(CCC(=C)Cl)=O)CCCC3)CCCCC1C2(F)F 67748,N1(C(C2CC(=C)C2)=O)CC2(CC(CNC(C3(CCOC)CC3)=O)C2)C1 67749,N1(C(Cc2cc(C)sc2)=O)CC(C)CN(C(c2ccc(N(C)C)nc2)=O)CC1C 67750,C1(NC(N(C)Cc2ccc(Nc3ccccn3)nc2)=S)CCC(F)(F)CC1 67751,c1(CCc2n(CCC=C)nc(-c3ccnc(Cl)c3)n2)ccc(C)c(C)c1 67752,c1(NC2CCN(CC)CC2)nc(N2CCC3(CCCN3C)C2)nc2sccc12 67753,c1(C(=O)NC(C2N(C(CCc3nc(C)sc3)=O)CCC2)C)cc(C)c(C)o1 67754,C1(CNC(Cn2ncc(CC)c2)=O)CN(C(=O)CSC(F)F)CCC1C 67755,CC1(C)C(NC(N2CCCC2c2ncc[nH]2)=O)CC1O.c12ccnc(n1)O2 67756,C(=O)(CC(C)CCC=C(C)C)N1CCCCC(CNC(C(C)NC(CC)=O)=O)C1 67757,CCC(C)C(=O)C(=O)N1CC(C(=O)NC2CCN(C3CC3)C2=O)C(F)(F)C1 67758,C1(NC(C(CN(C)C)O)=O)(CO)CCCN(C(=O)CCCC2CCCC2)C1 67759,c1(N(C(CC)=O)CC)ccc(O)c(C(N2CCN(C(=O)Cc3ccco3)CC2)=O)c1 67760,C1(C(=O)NCC2N(C(c3c[nH]c(=N)s3)=O)CCC2)CCN(CCF)CC1 67761,C#CCCC(C(=O)NCCCc1ccncc1)NC(c1cnc(OC)s1)=O 67762,c1(C(N2CCC(F)(C(=O)Nc3cccc(O)c3)C2)=O)ccc(Br)c(F)c1 67763,C=CCC(C)(CC=C)NC(C1CCCCN1C(=O)CN1CCCCCC1)=O 67764,N1(C(C2CCN(C(C3(COCC)CCCC3)=O)C2)=O)CCC(CC(C)O)CC1 67765,C1(C(=O)NC2CCCCN(C(c3ccc(F)cc3Cl)=O)C2)CCN2CCOCC12 67766,C1(NC(c2n(CC)ccn2)=O)COC2(C1)CN(C(c1c[nH]c(C#N)c1C)=O)C2 67767,N1(C(CNC=O)=O)CCN(C(CNC(=O)CC2CCC(=O)N2)C(F)F)CC1 67768,C1(N(C)C)CCCN(C(=O)C(O)C2CN(C(C3(O)CCCCC3)=O)C2)CC1 67769,CC1CCCCC1OC.C1CCCCCNC(=O)CC(=O)OCCC(=O)N1 67770,Cc1nnc2n1CC(C(=O)NCCCOCCNC(c1ccncn1)=O)C2 67771,C1(C(=O)Nc2ccc(OC)c(N3CCOC3=O)c2)Cc2ccc(F)cc2C1 67772,C1(NC(CCc2n(C)ccn2)=O)CCCCC1NC(=O)CCN1C(=O)CCC1=O 67773,c1(COC)nn(C)cc1C(=O)N(CCNC(=O)CN1CCC(C)C1)CC1CC1 67774,c1(C(=O)NCC(C(=O)NCC(COC)O)C)cnn2ccccc12 67775,N1(C(CC2ON=C(CC)C2)=O)CC(CNC(c2ccc(Cl)cc2)=O)C2(CCC2)C1 67776,C1(COC)(CNC(=O)C=CC(C)C)CCCN1C(=O)CCc1nnc(C(F)F)o1 67777,C1(CN(C(=O)CN2CC3C=CC2C3)C)C(C2CC2)CCN1C(=O)CC1CC(F)C1 67778,c1(C(N2C(C)CC(CNC(=O)CCc3cnn(C)n3)C2)=O)cc2ncccc2o1 67779,N1(C(CNC(C(CC)CC)=O)=O)CCC(NC(=O)Cc2ccc(Cl)cc2)C(C)C1 67780,c1(C(=O)NCCCN(C(CCSCC)=O)C(C)C)ccn2cc(C3CC3)nc2c1 67781,N1(C(C(CCOC)OC)=O)CCN(C)CC1C(=O)NCc1ccnc(O)c1 67782,c1(C(=O)NC2C(OC)CN(C(C3(C(N)=O)CCC3)=O)C2)c(F)ccc(F)c1F 67783,C=CC(C)(CCOC)C(=O)NCC(C)NC(=O)CCC1CCC1 67784,N1(C(C(COC)CC(C)C)=O)CCCC(C)(C)C1C(N1CC2(CC(O)C2)C1)=O 67785,CCS(=O)CCNC(=O)CC1(N(C)C(c2cccn2C2CC2)=O)CC1 67786,c1(NC(=O)Nc2ccc(C3(O)COC3)cc2)c(F)ccnc1F 67787,Cc1coc(C(=O)NC2CC(OCC(=O)NC3CC3(C)C(C)C)C2)c1 67788,N1(C(COC)=O)C(C)C2CC1C2NC(c1sccc1C1CC1)=O 67789,C1(NC(c2cn(CC)nn2)=O)CCC2CCN(C(=O)C(F)CC3CCOC3)C1C2 67790,Cc1[nH]c(=NCCc2ccc(C(=O)NC3CCC(C(C)C)NC3=O)o2)ccc1C#N 67791,N1(C(C2N(CC)CC2)=O)CCC(=CCNC(=O)CCCCN2CCOCC2)CC1 67792,N1(C(c2ncc(C)c(C)c2)=O)CC2CCC1CC2NC(c1cnsn1)=O 67793,C1(C(=O)NCC(C(=O)NC2CC(O)C2)O)Cc2nccn2C1 67794,Cn1nnc2c1CCN(c1nnnn1CC(C1CCCC1)OC(F)F)C2 67795,C1(NC(C(F)=CC)=O)CCN(C(c2ccc(C)cc2C(C)=O)=O)CCC1CO 67796,c1(CCN(C(=O)N)CCO)ccc(F)c(Br)c1.c1(N2CCOCC2)ncc(Br)s1 67797,N1(C(c2cnc(OC)s2)=O)CCC(C(C)NC(C2CCCOCC2)=O)CC1 67798,c1(C(=O)NC(C(C)NC(c2ccc(C(C)C)cc2)=O)CO)cc2occc2n1C 67799,C1(NC(c2cc(O)no2)=O)CN(c2ncc(-c3ccccc3)cn2)CC1F 67800,C(C(=O)N1CCCC1C(C)NC(=O)COC1CCC1)(C(C)C)SC 67801,CC1(C)OCc2c1n[nH]c2C(=O)NC1CC1NC(=O)Cc1cccnc1Br 67802,CC(CCC(=O)NC1CC1)NC(C1CCCN1C=O)=O 67803,N1(C(Cn2cc[n+](C)c2)=O)CC2CC2(NC(=O)CC2CC=CCC2)C1 67804,C(=O)(C=CS(F)(F)(F)(F)F)NCCN(C(CC(CC)(C)C)=O)CC 67805,C1(NC(C2C(C)C2C)=O)CN(C(C2CCC(C(N)=O)C2)=O)C2CCCC12 67806,N(C(=NCCc1cncnc1)NCc1ccc(=N)[nH]c1)C1C(C)C1 67807,C1(CC(N2C(CN(c3ccncn3)C)CCC2)=O)CCC2CC12 67808,N1(C(CCc2cncc(C)c2)=O)C(C)CN(C(C2C3CCC(F)(F)C23)=O)CC1C 67809,C(C)(CCC(F)(F)F)NC(CC1(NC(c2n(CC)c(O)nc2)=O)CC1)=O 67810,c1(NC(C2N(C(CCCC#C)=O)C3C(C2)C3)=O)c(C(=O)OCC)ccc(Cl)c1Cl 67811,CCN(OC)C(=O)C(C1CCCC1)NC(c1sccc1OC)=O 67812,c1(OC(C)C)ccc(C(=O)NCC2C=CCN2C(=O)C(F)C(C)C)nc1 67813,c1(C(=O)Nc2ccc(CN3CCC(c4ccccc4)CC3)o2)cc(O)cc(O)c1 67814,C(=O)(C(C)(C)C(C)(F)F)N1CCCC(C)(C(=O)NCC2C(C)(C)C2)C1 67815,Cc1[nH]nc(CO)c1C(=O)O.N1(CC(=O)NC(C(N)=O)C2CCCC2)CCCCC1 67816,c1(CS(N2CC(C)N(c3ncccn3)CC2)(=O)=O)ccc2c(c1)OCO2 67817,CCCC(CC(=O)NC1CCC(=O)NC1C)NC(=O)Cc1cnsc1 67818,CC1CN(C(C2CCN2C(C)(C)C)=O)CC1CNC(=O)C(c1ccccc1)O 67819,N1(C(c2ccc(N3CCCC3)cc2)=O)CCN(Cc2ccc(I)c(O)c2)C2CC12 67820,c1(C(=O)NCC(CNC(=O)CCn2ccc(C)n2)OC)cc(Cl)cc(F)c1N 67821,c1(C(=O)OC)cnc(C(=O)OC2CC(C(=O)NC(=O)C3CC3)C2)n1C 67822,C(=O)(CCCCCF)NCC#CCNC(c1cc(C#N)sc1)=O 67823,C1(C(=O)NCC(CNC(C(C)OCC)=O)OC)OCCN(C)C1=O 67824,C1(OC)CC(CNC(=O)Cc2cc(C3CC3)no2)N(C(C2CCC(F)(F)C2)=O)C1 67825,O=C(CC1COCCN1c1ncnc2n[nH]c(Br)c12)N=c1cc[nH]cc1O 67826,c1(C(=O)NCC(C)(CO)NC(C2C(F)(F)C23CC3)=O)nn(CC(F)F)cc1[N+](=O)[O-] 67827,CC1C(NC(=O)C2=COCCC2)CCCN1C(c1ncc(F)cc1N)=O 67828,N1(C(C2(C)CC2Br)=O)CCCC(n2cc(COCCOCCCO)nn2)C1 67829,n1(CC(=O)NC2(COC)CCN(C(=O)CNC(C)=O)C2)ncc2cc(C)cnc12 67830,C(CC(=O)NCCCCNC(c1cc(C)ccn1)=O)(C(C)C)OCC 67831,C1(OC)CC2(C1)CC2NC(=O)NOCCC(C)O 67832,N1(C(c2cnccc2Cl)=O)CCCC12CN(Cc1ccc(Cl)nc1Cl)C2 67833,C1(C(C)C)CN(C(=O)CCCn2cccc2)CCCN1C(=O)CS(C)(=O)=O 67834,c1(N(CCN(CC)CC)CC)ccc(S(=O)(=O)N(C(C)CC#N)C)c(Cl)c1 67835,c1(C(N(C(C)CNC(c2cnc(C)n2C)=O)CC)=O)cc(C)c2nc(C)cn2n1 67836,C1(NC(C(C)c2ccco2)=O)CCCC(NC(=O)C=CI)C1 67837,c1(C(=O)NCC2C(NC(CCCCOC)=O)CC2)cccc(O)c1C 67838,N1(C(C2(SC)CC2)=O)CCC2(CCN(C(c3ccc(C(N)=O)s3)=O)CC2)C1 67839,C1(NC(C(CC)F)=O)CCOC12CCN(C(c1nc(C)c(C)nc1C)=O)CC2 67840,O=C(CCCC(F)(F)CO)NC1CC2CCC(C1F)N2C(C1CC2CCC2C1)=O 67841,CC(O)C(C)(C)CNC(c1cc(CNC(=O)C(O)CCN(C)C)no1)=O 67842,c1(CC)nn(C)c(C(N2CCC(CO)(NCc3ccccc3Br)CC2)=O)c1Br 67843,C1(C)(CNC(c2c(CC)noc2)=O)CCN(C(=O)CC2CC2(Cl)Cl)C1 67844,CC(C)(C)C(=O)N1CCCC1NC(=O)NC(Cc1cncs1)C(=O)O 67845,CCCCCCC(C)C(=O)NC(CN(C(c1cn2c(n1)CCC2)=O)CC)CC 67846,c1(C(N2C(CNC(C=C(CC)C)=O)COCC2)=O)ccc(C)c(S(C)(=O)=O)c1 67847,C1(F)(CNC(CS(=O)(=O)N(C)C)=O)COCCN(C(=O)CS(=O)(=O)N(C)C)C1 67848,Cc1cc(Br)cc(Cl)c1NC(=O)NCc1nccn1C 67849,N1(C(C2(CC#C)CC2)=O)CCC(C(=O)NCC(=O)NC2CCCC2)C(C)(C)C1 67850,c1(C(C(=O)NC)N(C(C)CCO)C)ccc(Cl)c(C)c1 67851,c1(CC(=O)NCC23OCC(NC(CCSC)=O)(C2)C3)cc(Cl)ccc1Cl 67852,N1(C(C(C)C(F)(F)F)=O)CCCCCC(NC(=O)Cc2cn3ccsc3n2)C1 67853,N1(C(C2N(C(c3cn(C(C)C)nc3)=O)CC(O)C2)=O)CCCCC(CO)C1 67854,C(=O)(CC(C)(C)CNC(=O)Cc1cncc(C)c1)N1C(CO)CC(OC)C1 67855,CC1(CNC(C2CCNC2=O)=O)CCN(C(C2SCCCS2)=O)C1 67856,CCC(C)CCCCC(=O)NCCCCCN(C)C(C1(OC)CCC(C)(C)C1)=O 67857,C(=O)(C1=CCCOC1)NC1C(CC)N(C(c2cnc(CC(C)C)[nH]2)=O)CC1 67858,N1(C(CCC=CC)=O)Cc2[nH]nc(C(N3C(C)CCC3(C)C)=O)c2C1 67859,C1(NC(CCS(=O)(=O)NC)=O)(CNC(c2ncccc2C)=O)CC2CCC1CC2 67860,c1(OC)ccc(OCC2CC2)c(CC(=O)NCC2Cc3nccn3C2)c1 67861,C12(C(=O)NCc3ccc(COC)c(F)c3)CC3CC(C1)C(=O)C(C3)C2 67862,C1(OCC)CN(c2ccc(N3CCN(C)CC3)nn2)CC1c1nn[nH]n1 67863,N1(C(c2cccc(NC(C)=O)c2C)=O)CCCC12CN(Cc1ncsc1C)C2 67864,C1(C)(N(C)C)CCCN(C(C2(F)CN(C(=O)CCCF)C2)=O)C1 67865,N1(C(CNC(CNC(C)=O)=O)=O)CC2CC1CCN2C(c1ncc[nH]c1=O)=O 67866,c1(C(N2CC(CCc3cn(CC(c4ccccc4)OC)nn3)C2)=O)cnc(O)o1 67867,C1(CCNC(CCCC)=O)CCCCN1C(=O)COCc1scnc1C 67868,CCC(CC)C(C(=O)N1CCC(C(=O)N(CCCSC)C)(CC)CC1)OC 67869,CC1CCN(C(c2cnn(C)c2C(F)(F)F)=O)CC1NC(C1CC(F)(CO)C1)=O 67870,c1(NC(N2CC3(CN(C)C(=O)CC3)C2)=O)cc(Cl)c2cc(Br)ccc2n1 67871,c1(C(=O)NCc2c(C)cco2)ccnc(CNC(=O)COc2ccsn2)c1 67872,c1(CNC(C2CCC3(CC3)C2)c2n(C3(C)CC3)nnn2)cccc2sccc12 67873,c1(C(N(CC(CNC(COC(c2nccn2C)C)=O)O)C)=O)ncc(Cl)s1 67874,c1(C(CNC(=O)C(N2CC(O)(C(F)(F)CO)C2)=O)=O)cc(F)ccc1F 67875,c1(C(N(CCCCNC(C(C(COC)C)C)=O)C)=O)cnn(C)c1S(N)(=O)=O 67876,C1(C(=O)NC2(C)CN(C(=O)CO)C2)C2Cc3ccccc3C12 67877,c1(C(=O)NC(CC(C)NC(C2CC(=C)C2)=O)C)noc(-c2ccccc2)c1C 67878,CC(CC(=O)NC1COCC1C(=O)N(C)CC1CCCS1)N(C)C 67879,CCCC(CCC)C(=O)N(C1CCN(C(C2(CCOC)CCCC2)=O)C1)C 67880,c1(OC)ccc(CCC(N2CCC(CNC(=O)CSC)C2(C)C)=O)cc1O 67881,c1(NC2(c3n(CCOCC)nnn3)CC(C)N(C)C2)cc2c(cc1OC)CCC2 67882,C1(NC(=O)CC2CCCNC2=O)CN(C(=O)CSC2CC2)Cc2nccn2C1 67883,CC(C)C(C)(O)CNC(c1sccc1CNC(=O)C=Cc1cccnc1)=O 67884,Cc1nc2c(s1)CCCC2CN(C)C(c1cnccc1C1OCCO1)=O 67885,C1(C(=O)NC2(CCCNC(CSCC)=O)CC2)CC(C)CC(C)C1 67886,C#Cc1cn(C)nc1C(N1CCC1CNC(c1cccc(O)c1C)=O)=O 67887,c1(C(=O)NCCCOCCC(=O)N(CCCC)CCCO)cc(C(C)(C)C)n[nH]1 67888,n1(CC(N2CC(C)(NC(CC=C)=O)C2)=O)cc(C)c(O)nc1=O 67889,C(=O)(CCC(C)(C)F)N(CCC(=O)N(CCC(C)O)C)CCO 67890,C(=O)(CCCCC(C)C)NC1CC(CNC(C(CC)NC(C)=O)=O)OCC1 67891,N1(C(CCCOC)=O)CCN(C(=O)CCc2nnc(S)nc2O)CC12CC2 67892,C1(NC(c2ccn(C)n2)=O)CN(C(=O)C(F)C2CCOC2)CC12CCCC2 67893,C=CC1CCCN(C(c2ccc(CNC(=O)CN(C)CCOC3CC3)nc2)=O)C1 67894,CCCCC(C)(F)C(=O)N1CC(CC(F)C(=O)N(C2CC(O)C2)C)C1 67895,N1(C(c2ccc(SC(c3ccccn3)COC)o2)=O)CC(C(=O)NC)C2(CC2)C1 67896,Cc1cc(N(C(=O)CC2(NC(c3cnc(S)nc3)=O)CC2)C)cc(C)c1 67897,c1(C(N2CC(CNC(C3(Cl)CC3)=O)C(O)C2)=O)cc(F)c(C(F)(F)F)c(F)c1 67898,C=CCC(CC)C(=O)NC(CNC(=O)C(O)CC1CCCC1)CCCC 67899,C1(N(C(=O)C(C)(N)C(=O)O)C)CC2CCCC1N2C 67900,CCCC(C)CC(=O)NCC(C)(CC)C(=O)NCc1cc(C(C)C)no1 67901,n1(CC(=O)NCC(C)CNC(c2nc(Cl)cs2)=O)nnc(-c2ccccc2)n1 67902,CC(Cc1cnc[nH]1)C(=O)N(C1CCN(C(C2CC(F)(F)C2)=O)C1)C 67903,c1(OC)ccc(C(=O)NC(CNC(=O)CC(C)(C)C#N)C(C)(C)C)cc1F 67904,c1(C(=O)NCCCN(C(C(C)OCCC#C)=O)C)c(OC)ccc(F)c1Br 67905,CC1(C)OCCC1C(N1CC(OC2CCN(C(=O)COCC3CC3)CC2)C1)=O 67906,c1(C(N(CCCNC(=O)CC2(C)CC2F)CC)=O)cnc(SC)nc1O 67907,N1(C(c2c(CC)cccc2)=O)CCCC(C)C1CNC(=O)CC1CCS(=O)(=O)C1 67908,C1(CNC(c2nc(CCC)sc2)=O)CN(C(c2nocc2Cl)=O)CCC12CCC2 67909,C1(C(=O)NCC=CCNC(COC(C)C)=O)CCCC(C2CC2)O1 67910,N1(C(CC2N(C(c3ccc(O)cc3)C)CCOC2)=O)CCOC(C(C)(C)C)CC1 67911,c1(C(C)C)ccc(CN2CCN(C(=O)Cn3cncc3CCN(C)C)CC2)cc1 67912,C(CC(=O)NC1CCCC2(C1)N=N2)(C(F)(F)F)NC(C(CC)=CCCC)=O 67913,C(C1CCCN1C(=O)CC1CC2CC2C1)=CC(N1CC(C)(C(=O)OC)C1)=O 67914,c1(C(=O)NC2C3(CCN(C(CCC)=O)C3)CCC2)ccc2ccc(Br)cc2n1 67915,N1(C(C2(C)C(C)OCC2)=O)CCC(CNC(C2(c3ccno3)CC2)=O)C(O)C1 67916,C(CCCC(=O)N1CCOC(CCO)C1)NC(C(C=C)O)=O 67917,c1(CNC(c2c(CNC(C3C(CCC)C3)=O)c[nH]n2)=O)ccnc(F)c1F 67918,C1(C(N2C(C(=O)OC)CC2)=O)CCC(NC(c2cc(C(C)=O)on2)=O)C1 67919,c1(-c2cn(C(CNC(C3C(=C)C3)=O)C)nn2)cccc(Cl)c1Cl 67920,S(=O)(=O)(c1cccs1)NC(C)C(=O)NCC(=O)Nc1cc(F)ccc1O 67921,C1(CNC(Cc2scc(C)n2)=O)CN(C(=O)C(F)(F)C(F)F)CCC1(C)C 67922,C1(OC)COCCC1CC(=O)NCC(C)(C)CNC(c1scc(C)c1Cl)=O 67923,C1(CNC(CSSC)=O)CN(C(=O)C(C)c2ccco2)CC1C 67924,CC(CN(C)C)CC(=O)NC(C)(C)C(=O)NC1CC(=O)N(C(C)(C)C)C1 67925,C1(NC(c2ccc(Cl)o2)=O)C2CN(C(=O)Cc3ccccn3)CC12 67926,C(c1ccc(OCC(O)CSC2CC3(CC3)C(=O)O2)c(OC)c1)=CC 67927,N1(C(CN(CCCCCC)C)=O)CC2CC1C2CNC(=O)CC(C)(C)O 67928,c1(OCC)nc(C(=O)NC2(C(=O)NC3CC(C(N)=O)C3)CC2(C)C)co1 67929,CC(C)C(CNC(c1ccnn1C)=O)NC(c1cc(-c2ccco2)[nH]n1)=O 67930,N1(C(C2=CC(C)(CC)C2)=O)Cc2ccccc2C(NC(C2(F)CCCC2)=O)C1 67931,CC1CN(C2CCCN(c3ccccc3OC(F)F)C2=O)S(=O)(=O)C1 67932,N(C)(C1CCc2ccccc21)CC(C)NC(Cc1ccc(OC)cc1Br)=O 67933,C1(C(N2C(C)(C(C)C)CC2)=O)CCCN(C(=O)C(C)CC2CC2)C1 67934,c1(C(N(CC(C)N(C)C(C2CC2CF)=O)C)=O)ccc2c(c1)C(=O)CCS2 67935,C1(C2CC2)(CNC(CC2C(C)(C)CC2)=O)CCN(C(c2ccc(Cl)cc2O)=O)C1 67936,C1(NC(c2ccn(CCCC)n2)=O)CN(C(=O)CCn2cccnc2=O)CC1O 67937,c1(OC(=O)CSCCC(=O)N2CC(NC(=O)C(O)C3CC3)C2)ccccc1Br 67938,c1(CN2C(C(=O)Nc3ccc(-n4cccn4)nc3)CC(O)C2)ccc(Br)cc1O 67939,C12(CNC(C3C(C=C)CC3)=O)CCC(CC1)N(C(C1CC3CC3C1)=O)C2 67940,C(=O)(CC1CCc2ccccc21)NC1CC(O)(CNC(c2cc(C)c(C)o2)=O)C1 67941,C1(C(=O)NCC2CCC(O)C2)CC2CC2N1C(=O)CO 67942,c1(CC(=O)NC2C(NC(C3(C(N)=O)CC3)=O)C2)ccc(Br)cc1Cl 67943,C(=O)(CC(C(F)F)C(C)(C)C)NC(CNC(c1c(N(C)C)cccn1)=O)C1CC1 67944,c1(OCC)ncccc1C(N1CCC(C)C1C(=O)NOCc1ccncc1F)=O 67945,N1(C(C=CCC)=O)CCN(C(=O)CNC(N)=O)CC1CC 67946,c1(NC2C(NC(C(C)SCC)=O)CCCC2)ncnc2cnccc12 67947,c1(C(=O)OC)c(N2CCC(CNC(=O)C(C)C3CC3)C(C)C2)ncnc1Cl 67948,C1(CC=C)(NC(=O)Cc2cccc(Cl)c2)CCCN(C(c2cocc2C)=O)C1 67949,C1(CNC(C2CC(C)(C)OC2)=O)CC2CCC(C1)N2c1cnc(C(=O)ON)cn1 67950,c1(N(C)CC2CCCN2C(=O)CC2CCOCC2)ncccc1S(C)(=O)=O 67951,C1(c2n(C)nnn2)(NCCOCC2CC2)CC2COC1C2 67952,C(=O)(CC1=NNC(=O)C1)NC1CCN(CCNC(C2(C=C)CCC2)=O)CC1 67953,c1(C(=O)NCC2CC(O)(CNC(C(C(C)C)O)=O)C2)cscc1S(C)(=O)=O 67954,C(C)(C(C)(C)C(=O)NC1C(C)(C)C1(C)C)NC(c1ccc(CC)[nH]1)=O 67955,N1(C(c2c(C)snc2)=O)CCC2CCN(C(c3cc4n(c3)CCCC4)=O)C2C1 67956,CC1Cc2cccc(C(=O)NC3(CNC(c4ccc(F)cc4)=O)CCC3)c2O1 67957,N1(C(Cc2cccc(C)n2)C)CCC(O)C(C(=O)NC(c2cccc(F)c2)C)C1 67958,C1(NC(=O)Cc2c[nH]nc2O)C=CCN(C(C2(F)CC2c2ccccc2)=O)C1 67959,C(CN=c1[nH]c(=NC(C)c2cc(C)on2)[nH]c2c1SCC2)SCCOC 67960,CCC(O)CC(=O)N1CC(CF)(NC(c2cccc(C(F)F)c2)=O)C1 67961,N1(C(c2n[nH]c(C)c2C)=O)CCCC12CCCN(C(C1CCCCC1(F)F)=O)C2 67962,C1(NC(c2c(C)nc(N(C)C)s2)=O)CN(C(=O)C=CC(=O)N(C)C)CC1C1CC1 67963,C(=O)(CCC(C)(C)c1ccccc1)N(C1CCCC(O)C1)CC 67964,c1(C(=O)NC2CN(C(c3c(CC)non3)=O)C(C)CC2)cnc(O)c([N+](=O)[O-])c1 67965,C(=O)(C1=CC(O)C(C(=O)O)C1)N1CCC(C(C)NC(=O)CN2CCS(=O)CC2)CC1 67966,c1(C(=O)NC(CCNC(CCSC)=O)(C)C)cn(C)c(-c2ccccn2)n1 67967,C(N=c1cc(Cl)nc(C(C)OC)[nH]1)C1N(C(c2nc(CC)oc2)=O)CCCC1 67968,N=c1c(-c2noc(-c3ccc4nc(O)[nH]c4c3)n2)c[nH]c2ccccc12 67969,N1(C(=O)CC2CN(C(=O)CC3CC4CC4C3)CCO2)CCc2nn[nH]c2C1 67970,CCS(=O)C1CCCCC1NC(=O)C(=O)N(C1CCOC1)C 67971,N1(C(CCC#CC)=O)CCN(C(=O)C=C(C)C(C)C)CC2CCCCC12 67972,N1(C(c2cn(CC=C)nc2)=O)CCC2(CCN(C(=O)C(F)=C3CCCC3)C2)C1 67973,C1(CNC(CC(=O)OC)=O)CN(C(=O)C(n2nccc2C)C)CC12CCC2 67974,C(=O)(C(O)C1CN(C(c2ccoc2)=O)C1)NCC(=C)Cl 67975,c1(-n2cc(CNCc3cccc(F)c3)nn2)ccc(Br)c(Cl)c1F 67976,c1(C(C(=O)NCC(=C)CCNC(C2CC(C)(F)C2)=O)(C)C)cccc(C)c1 67977,c1(C2(NC(=O)Nc3cc(C)ncc3)CC2)cc(F)ccc1F 67978,C1(C(=O)NC(C(=O)NCC(C(C)C)(C)F)CCC2CCC2)CC2(CCC2O)C1 67979,C(=O)(CC1=CCOCC1)N1CC(C)(C)C1C1CCN(CC(C(=O)C(F)(F)F)=O)CC1.OC 67980,N#Cc1ccc(CNC2CC(C(=O)Nc3cncc(F)c3I)C2)c(Br)c1 67981,c1(C(N(C2CCN(C(C3CC3(F)Cl)=O)CC2)CC)=O)cc(Cl)cc(Cl)c1N 67982,C1(NC(Cc2scc(OCC)n2)=O)CC2(C1)CN(C(=O)CC#N)C2 67983,c1(NC(C2CCN(CCC(O)CO)CC2)=O)cnc2ncc(-c3cscn3)cn12 67984,C(C(C(=O)NCC1(F)CC(CO)C1)N(C)C)NC(C1C(C)CC1)=O 67985,c1(-c2cn(CC3(C)CCC3)nn2)nc2ccccc2s1 67986,CC1CCC(NC(c2nc(Cl)ccc2F)=O)CN1c1ncc(F)cn1 67987,CCCCCCC(CC)(CC)C(=O)N1CCC(N(C(=O)C(F)C(F)(F)F)C)C1 67988,N1(c2ccnc(NC3CC(C)N(C4CC4)C3)n2)CC(S(N)(=O)=O)C1 67989,CC(=O)N1C(=O)C(c2cccc(C(F)(F)F)c2)N1C(=O)CC=C(C)C 67990,c1(C(N(CC(CNC(c2nc(C)sc2C)=O)C)C)=O)cc(N)cc(O)c1C 67991,C(=O)(C1=Cc2ccc(Cl)cc2OC1)N(C1CCN(C(C2CC(=O)NCC2)=O)C1)CCO 67992,c1(OC)ccc2c(c1)CC1(CC1)N(C(C1C3CC(N)CC13)=O)C2 67993,C(=O)(CC(O)CC(C)C)N(C1CCN(C(c2c(C)cccc2Cl)=O)CC1)CCO 67994,C(=O)(Nn1cnnc1C)C1N(CC)CCCC1.C1CCC(=O)O1 67995,CCC(C)CCCCC(=O)N(CCN(C)C(C1CC2CCC1C21CC1)=O)C(C)C 67996,C1(C(=O)NCC(C)Cn2cccn2)CC(=O)CN1C(C1OCCC1(C)C)=O 67997,N1(C(C(C2CC2)OC)=O)CCC(CNC(=O)CCCN=[N+]=[N-])C(C)C1 67998,c1(C(=O)OCC)cn(C)nc1NC(=O)CCN(CC(C)C(C)C)C 67999,N1(C(CN(CC#C)C(C2CN3CCN2CC3)=O)=O)CC2CC(N(C)C)C(C2)C1 68000,c1(CC)cc(C(=O)NCC(C)N(C)Cc2cccc(Cl)c2F)cc(O)n1 68001,C1(C)(C(N2CCCC(CN(C(=O)C=CC=C(Cl)Cl)CC)C2)=O)CCC(=O)CC1 68002,C(=O)(CC(C(F)F)NC(=O)Cc1ccns1)NCC(C)SC 68003,Cc1ccc(-c2cc(C(=O)NCCCCC(C)NC(=O)CC(C)(C)F)on2)cc1 68004,c1(OCCC=C)cccc(CC(=O)NCC2CC2CNC(=O)CCOC)c1 68005,Cn1cncc1CC(N1CC(O)(C(C)(C)CNC(C2CC2F)=O)C1)=O 68006,c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)CC2C)cncn(C)c1=O 68007,C1(C(=O)NC(C2CCCC2)CNC(COCCCCC)=O)CCN(C2COC2)C1 68008,c1(C(=O)NCC(CNC(C(F)=C(C)C)=O)(C)O)c[nH]nc1[N+](=O)[O-] 68009,CCCC(C)(C)C(=O)NC1CCCC(CNC(=O)CC2(CS(C)(=O)=O)CC2)C1 68010,c1(C(CNC(=O)CC2CC(C)(C)C2)NC(c2c(C)snc2)=O)ccc(F)cc1F 68011,Cc1cc(C(N2CCCC2c2nc(-c3ccccn3)cs2)=O)c(C)n1C(C)C 68012,CC(C)C(F)C(=O)NC12CC1CN(C(c1cnn(C)c1CN1CCCC1)=O)C2 68013,N1(C(c2onc(C)n2)=O)CCN(C(=O)COCc2ccccc2F)C(CCO)C1 68014,c1(CNC(C2CCC(C(N)=O)O2)=O)ccc(-c2ccccc2)nc1 68015,C1(NC(C(C(C)C)n2cnnc2)=O)CCN(C(c2n[nH]cc2Cl)=O)CC(O)C1 68016,C1(NC(C2CCC(=O)C2)=O)CN(C(c2scnc2C(F)F)=O)CC12CCOCC2 68017,C(=O)(C#Cc1ccc(Cl)cc1)N(c1c(C)c(N(C)C)ccc1)C 68018,c1(OC)cc(C)c(CN2CC(C(=O)OC)CC2CO)cc1NCC1CCCO1 68019,C1(NC(c2coc(Br)c2)=O)CCC2CCN(C(=O)CCC3CCCO3)C12 68020,CC1=C(CNC2CN(Cc3ccccc3)C(C)(C)C2)SCCO1 68021,c1(C(=O)NCC2(C)CCN(C(C3C(C#C)C3)=O)CC2)cc(C)c(F)cc1F 68022,c1(C(N2C(CNC(C(C)OC3CCCC3)=O)CC2)=O)ccc(O)cc1[N+](=O)[O-] 68023,N1(C(Cn2c(C)nnn2)=O)CCN(C(=O)COc2ccc(O)cc2)C(CCO)C1 68024,C1(C(=O)NCC(=O)OCCCC)CC(O)CN1C(c1ccn(C(F)F)n1)=O 68025,C(=O)(C(C)(C1CCC1)NC(C1CCN(C)C1)=O)NCC(C1CCC1)OCC 68026,N1(CC=C)C(=S)NC(c2csc(C3CCCCC3)n2)C(C(=O)NCCC)=C1C 68027,CC1CN(C(=O)CCC(F)(F)F)CC1(C)CNC(=O)CC1(C)CCC1 68028,C12(OCC)CCC(C(N3CCC(CF)(NC(=O)CSCC(N)=O)C3)=O)(CC1)C2 68029,N1(C(C=CC=CCC)=O)CC(=O)NCC1C(N1CC(O)(CCC)C1)=O 68030,N1(C(COCCOCCOC)=O)CC(CCC2CCC3CC23)(C)C1.C(=O)OC 68031,c1(C(N2CCC(C(C)(C)NC(CC(C)SC)=O)CC2)=O)n[nH]c2c1CCCCC2 68032,c1(OCC)ccc(OC(C)C(=O)NCCc2oc(C)cc2C)cc1 68033,C1(COC)C2CC3CC(C2)CC1C3.C12(CCCC(C)C1)c1nnnn1CCN2 68034,c1(C(N2CCC(N(C(=O)CN3CCC3C)CC#C)CC2)=O)ccc(O)c(F)c1 68035,C12(NC(C(c3c(C)cccc3Br)NC(C(CSC)O)=O)=O)CC1COC2(C)C 68036,Cc1nn2cc(C(=O)NC3CC(C(=O)NCCC4CCC(C)O4)C3)nc2s1 68037,C1(O)(CC)CCN(C(C2C(NC(=O)Cc3cc[nH]c3)C2(C)C)=O)CC1 68038,C1(C(N2CC(CC#C)OCC2)=O)CCN(C(C2CC23CCOCC3)=O)C12CCC2 68039,C1(N(C(=O)NC2CN(CC)C2)C)CCCN(C(c2cc(C)oc2C)=O)C1 68040,C(CC(=O)NCCS(C)(=N)=O)(CC(C)C)NC(c1c(C)cc(C)nc1)=O 68041,C(=O)(CC(O)C(C)(C)C)N1CCC(F)(CNC(c2c(C)n(C)nc2)=O)CC1 68042,C=CCC(CC)C(=O)NC1(CCOC)CCN(C(=O)CC2(O)CCCC2)C1 68043,c1(C(=O)NCC2(C)CCC(NC(C=C(C)C(C)C)=O)C2)ccc2cc[nH]c2n1 68044,CCC(C(=O)N(CCCN(C)C(c1cc(O)cs1)=O)C)OC1CCCC1 68045,C(=O)(C(C)(C)N(C)C)N1C(C(=O)NC(C=C)C2CCC2)CC1 68046,N1(C(C2C(C)CC2)=O)CCC(CO)(CNC(C2CC(n3cnnc3)C2)=O)CC1 68047,N1(C(COC2(C)CCC2)=O)CC(NC(=O)Cn2cc([N+](=O)[O-])cn2)C2(CC2)C1 68048,C1(CNC(C=C(CNC(C=CC(C)(C)SC)=O)C)=O)CCOC(C)C1 68049,C(=O)(C1=CC2(CCOC2)C1)N1CC2C(CNC(c3c(C)nncc3)=O)C2C1 68050,N1(Cc2c(OC(C)C)ccc(Br)c2)CC2CCN(C(c3cc[nH]c3)=O)C2C1 68051,c1(C(N2C(C)CCC(NC(c3csc(C#N)c3)=O)C2)=O)ccn2nccc2c1 68052,c1(OC)cc(OC)c(N)c(C(N2CCC(C(C)NC(c3ncccn3)=O)C2)=O)c1 68053,C1(CNC(C(c2cccc(F)c2)C)=O)CN(C(C2CC(=O)C2(C)C)=O)CCCO1 68054,Cc1cnc(C)c(C(=O)NC(CNC(C2COC2)=O)CC(C)C)c1 68055,N1(C(c2ccc(-c3csc(C)n3)s2)C(=O)NC)CCCN(C2CCC2)CC1 68056,Cc1ccncc1C(N1CCC(N(CC(N2CCC(C(=O)N(C)C)CC2)=O)C)C1)=O 68057,c1(OC)ccc2c(c1)OCC(C(=O)NC(CNC(c1ccc(C)s1)=O)CO)C2 68058,CC(C)CN=C(NCC(C)(C)C(C)(C)C)N1CCC(C)(F)C1 68059,n1(CCC(=O)N(C(C)CNC(=O)Cc2cnsc2)C)cnccc1=O 68060,c1(C(N2CCC(NC(C(C3CCC3)OCC)=O)C2CC)=O)cc(N)ccc1O 68061,CCC(C(=O)NCC1(NC(=O)CCc2cccnc2)CCC1)C(C)C 68062,C1(CNC(Cc2cc(C)sc2C)=O)N(C(=O)C(C)CC(C)C)CCC1(C)C 68063,C(=O)(CCC(F)(F)C(F)F)NCCCNC(CCc1nc(C)sc1)=O 68064,c1(CC)ccc(C(=O)NC(CNC(C2CC2(F)F)=O)CC)cc1[N+](=O)[O-] 68065,c1(OC)cccc2c1C(C(=O)NCC1CC1NC(c1ncccc1OC)=O)CC2 68066,C12(CCN(C(C3C4CC5C(C4)C35)=O)CC1)CN2.C(C)(C)(C(=O)NCC)OC(C)=O 68067,CC(C(=O)NC1CC(CNC(=O)C=CC2(C)CCOCC2)CC1O)S(N)(=O)=O 68068,C(=O)(CCCCCOC)NC1CN(C(CC(CC)OC)=O)CC1O 68069,CC1(C(=O)NCC2CCN2C(C2CCCCS2)=O)CC2(CCC2)C1 68070,O=C1CCC(O)CN1Cc1cn(CC2CCN2)nn1.c1(C2CC2)cccnc1 68071,CCC(C)CC(C(=O)NCCCn1cc(C)cn1)NC(c1cnc2n1CCC2)=O 68072,C(N=c1[nH]cnc(Cl)c1Br)C1(CNC(CCCC(C)C)=O)CC12CCC2 68073,C12(NC(c3cc(Br)co3)=O)CCCN(C(c3cc4cccnc4[nH]3)=O)CC1C2 68074,N1(C(CN(C)C)=O)CCC12CN(C(=O)CCc1ccc(Cl)cc1Cl)C2 68075,CC(C)CC(O)CC(=O)NCC1(O)CC(CNC(c2csc(CO)n2)=O)C1 68076,C1(C(=O)NC(CNC(COC(C)(C)C)=O)C2CCC2)CC2(C1)CC21CCC1 68077,N1(C(C(C(C)C)O)=O)CC2(C1)SCCC2NC(c1ccc(-n2cncn2)nc1)=O 68078,C1(C(=O)OC)(NCCN(C(C)Cc2sccc2Cl)CC)CCCCC1C 68079,CCC(C(=O)N(C)CCOCCCN(C(=O)C(C1CCCCC1)OC)C)OC 68080,C1(CNC(=O)CCN2CCC2)CC(O)CN1C(=O)CCc1csnn1 68081,C1(C(=O)NCC2(F)CCC(NC(CCCC#CC)=O)C2)CCCCC12OCCO2 68082,CCC(O)C(=O)N(C)CC1CCN(C(=O)CCNC(c2ccoc2)=O)C1 68083,C(=O)(C(C)C(O)CCCC)NC(C(=O)N1C(CC=C)CCCC1)CCCC=C 68084,c12ccnc(c1)C(=O)N2.c1(CC)n[nH]cc1C(=O)N(C(C)CN(C)C)CC 68085,N1(C(CCc2cnn(C)n2)=O)CCC2CCCN(C(=O)C=Cc3ccsc3)C2C1 68086,N12CCC(C3(CC3)C(=O)N1)CC2.C12(c3nnc(N4CC(C=C)C4)o3)CCOC(C)(C1)C2 68087,C=C(C)C1OCCC1N=c1nc2c(ncn2C)c(NCC2CCCC2)[nH]1 68088,c1(CC(=O)NCC(c2ccccc2F)NC(CC=C=C)=O)cn(C)nc1C(F)F 68089,c1(OC)ccc(C(=O)N(CCCN(C)C(c2sccc2Cl)=O)C)nc1OC 68090,C=C1CCN(C(c2cccs2)=O)C(C(=O)NCc2cc(C)ccc2O)C1 68091,C#CCC(C)C(=O)N(CC(C)(C)NC(c1cn(CC2(CC)COC2)nn1)=O)C 68092,c1(OCC)cc(Cl)ccc1C(N1CCN(C)C(CNC(=O)C(C)(O)C(C)C)C1)=O 68093,c1(C(=O)OCC)cc([N+](=O)[O-])c(NC(C)CCCNC(c2cnn[nH]2)=O)cc1C 68094,C#CCC(O)C(=O)N1CC(C(=O)NCCc2ccn(C)n2)C(CC)C1 68095,CCCCC(CC(=O)NCC(C)(O)C(C)CC)NC(c1ccccn1)=O 68096,C1(O)(CNC(=O)CCCn2ccnn2)CCCN(C(c2cc(O)nc(O)n2)=O)C1 68097,N1(C(c2cc(C)[nH]c2)=O)CCCC(O)(CNC(c2c[nH]cc(F)c2=O)=O)C1 68098,c1(CCC(N2CC(N(C(CC=C=C)=O)C)C(O)C2)=O)ccc(F)cc1Br 68099,c1(C(=O)NCCC(C)CCNC(C2COCCOC2)=O)cc(Cl)c(F)cc1O 68100,c1(C(N2CCCC(NC(c3c(OC)oc(C)n3)=O)C2)=O)c(C)cc(C)cc1C 68101,CC1(CNC(c2cc(Br)c[nH]2)=O)COCCN(C(c2cc(C#N)c[nH]2)=O)C1 68102,c1(C(C(=O)NC2CC2)N(C(CC)C(=O)OC)C)cnc2ccnn2c1 68103,c1(C(=O)NC(C(C)C)CNC(=O)Cc2ccccc2F)ccc2[nH]ccc2n1 68104,CC1(C)CCCCC1=CC(N1CCC(CCNC(=O)C2=COCCC2)C1)=O 68105,C1(NC(C2CC(OC)CN2C(=O)C(C)Cn2cccn2)=O)CCC(C2CC2)CC1 68106,C1(NC(COc2c(C(C)C)cccc2)=O)CCN(C(=O)CC2CCCO2)CC1C 68107,C1(c2nnnn2Cc2ccco2)(NCc2n(CCC)ccn2)COCCOC1 68108,c1(C(N2C(C)(CNC(COCC)=O)CCC2)=O)ccc(=O)n(C)n1 68109,C=CCCN=C(NCC1CN(C(N)=O)C1)N1CCC(c2nncs2)C1 68110,C1(NC(Cc2scc(C)n2)=O)CC(NC(=O)Cc2ccn(C)n2)C12CCOCC2 68111,c1(C(N2CCN(C(C3C(OC)CCCC3)=O)CC2C)=O)ccc(S(C)(=O)=O)s1 68112,N1(C(CCC2(C)CC2(F)F)=O)CCC12CCNC2=O 68113,c1(-c2nc(NC(=O)Nc3ccncn3)sc2)ccccc1I 68114,C1(C2CCN(C(=O)Cc3cccnc3N)C2)(NC(c2c(C)nc[nH]2)=O)CC1 68115,C1(C)(C(=O)NC2CC(N(C)CC)C2)CCCN(C(c2cc(C3(C)CC3)on2)=O)C1 68116,Cc1ccc(CC(=O)NC(C)(CNC(C2CCC(C)O2)=O)C2CC2)c(Br)c1 68117,C1(CC(=O)NC2(CCOC)CC2)CC2(CC2)CN1C(=O)CC1CCC=CCC1 68118,C1(NC(Cn2c(C)nc(C)n2)=O)COC2(CCN(C(c3nnn(C)c3C)=O)C2)C1 68119,C(N=c1[nH]c(N2CCC3CC3C2)nc(=N)[nH]1)C1(SC)CC1 68120,C(=O)(C1=Cc2ccccc2C1)NC1C2(CCN(C(CCSCC)=O)C2)C1 68121,C(c1ccc(-c2ccccc2)cc1)=CC(=O)NC1CC(NC(C=CS(C)=O)=O)C1 68122,C(=O)(C1CCCc2ncccc21)N1CCCC(NC(C(CC(C)C)OC)=O)C1C 68123,C1(NC(c2cnc(Cl)s2)=O)CCN(C(c2ocnc2C2CC2)=O)CCC1(F)F 68124,N1(C(C(CC)(C)O)=O)CC(N(C)C(c2cc(C)c(Cl)cn2)=O)C2(CC2)C1 68125,C=CCCN=C(NCc1ccc(CS(C)=O)cc1)NCC1CCCCC1 68126,N1(C(c2c[nH]c(=NC)o2)=O)CCC2(CC2C(N2CCC(C)CC2)=O)C1 68127,CC1(CNC(C2CCCCN2C(N)=O)=O)CCN(C(=O)C2=CCCSC2)CC1 68128,c1(CCC)c(C(=O)NC2CCCC2NC(=O)CN2C(=O)CNC2=O)cnn1C 68129,N1(C(COCCC)=O)C2CCC(C(N3CC(OC)C(OC)C3)=O)C1CC2 68130,C1(c2nc(C)on2)CCCN(C(C2CCCCCC2)C(=O)NC2CCC2)C1 68131,C(=O)(NNC(=O)C(N)c1cccc(I)c1)c1ccc(OC)c(Cl)c1 68132,N1(C(CC(CC#C)NC(=O)CC(C)COC)=O)CCn2nccc2C1 68133,N#Cc1ccccc1C=CC(N1CC(NC(=O)CCc2ncc[nH]2)C(O)C1)=O 68134,Cn1nc2c(c1NC(C1CSCCN1Cc1cc(F)ccc1F)=O)CCC2 68135,N1(C(C(C2CC2)OC)=O)CC(O)(C2(CNC(C3(Cl)CCC3)=O)CC2)C1 68136,C(=O)(C1=CC(C)(CC)C1)NCC(CN(C(=O)Cn1cc(C)cn1)CC)(C)C 68137,C(CCCCC(=O)N1CC(NC(=O)C=Cc2ccccn2)C(C)C1)=CC 68138,C1(O)(CN(C(C2(OC)CC2)=O)C)CCN(C(C2CCCOC2C)=O)CC1 68139,C1(CNC(CC(C=C)C)=O)CC2CCC1N(C(c1sc(Cl)cc1Cl)=O)C2 68140,C(=O)(CCCC(F)F)NCC1CN(C(C2CCCN(S(CC)(=O)=O)C2)=O)C1 68141,C1(NC(C2C(C)(C)N(C(c3cc(Cl)ns3)=O)CC2)=O)CCCOC12CCC2 68142,C(C)(c1cccnc1)=CC(=O)NCCN(C(=O)C(F)C(F)(F)F)CCC 68143,S(=O)(=O)(c1[nH]c(=NCc2c(C)cccc2Cl)ccc1Br)NCCOC 68144,C(=O)(CC(=O)N1CCC(N(C(=O)C(C2CCCC2)OC)CC)C1)NCC#C 68145,C(=O)(CN=c1ccc(C#N)c[nH]1)N1CCCC(N(C(C(CCC)C)=O)C)C1 68146,C(=O)(CC(F)(F)C(F)(F)F)N1C(C(C)NC(c2cncs2)=O)CCC1 68147,CCC(CC(=O)NC1CC(CNC(c2cnns2)=O)C12CCC2)CC(C)C 68148,CC(CCNC(c1cc(Br)n[nH]1)=O)CCNC(C1CCS(=O)CC1)=O 68149,CCCCC(C)CCC(=O)NCC1CCC(C(=O)NC(C2CCCC2)C)O1 68150,O=C1COC2CCN(C(c3cccc(C(F)(F)F)n3)C(=O)NC3COC3)CC2N1 68151,C1(F)(CNC(C2(C)C(C)C2)=O)CCC(NC(=O)CCc2ncc(F)cn2)C1 68152,N1(C(C(C)N(C(C)=O)C)=O)CC=CC(C(N2CCC2(C(=O)O)C(=O)O)=O)C1 68153,Cc1c(C(=O)NC2(c3ccccc3)CCN(C(=O)C(C)(Cl)Cl)C2)nnn1C 68154,C(CC(C)C)(C(=O)NC1CCN(C(c2c[nH]c(Br)c2)=O)C1C)OC 68155,C1(CCC)(NC(c2ccc(CO)o2)=O)CCCN(C(c2cccc(C)n2)=O)C1 68156,C1(NC(C)=O)CCN(C(=O)CN)C1C(N1CCCC1)=O.c1(C(=O)OC)ccoc1C 68157,c1(C(N2Cc3cc(F)ccc3C2)C(=O)NCCCC)ccc2ncccc2c1 68158,C(C(CNC(C1(CC(C)C)CCC1)=O)OC)NC(C1C(CCC)C1)=O 68159,N1(C(C(CC2CCC2)NC(c2ccco2)=O)=O)CCC(C(F)F)CC1 68160,C1(C)(NC(C2C(C(=O)NCC#C)C2)=O)CCN(C(c2oc(C)nc2CC)=O)CC1 68161,CC(C)C(CCNC(=O)C(N)=O)NC(=O)C(C(C)O)c1ccccc1 68162,CC1CN(C(C2(F)CCOCC2)=O)CCC1N=c1[nH]c(Cl)ncc1Br 68163,c1(C(N(C2CC(NC(c3cnc(=N)[nH]c3)=O)C2)C)=O)cccc(F)c1C(F)F 68164,C1(NC(CCN(CC#C)C(C2CC(C)(F)C2)=O)=O)CC2(CC2)C1 68165,S(=O)(=O)(c1ccccc1F)NCCC(=O)NC1C(CNC(C=CC(C)C)=O)C1 68166,c1(-c2c(C(=O)NC3CCN(C(C=CCN(C)CC)=O)C3)nco2)ccccc1F 68167,CC1=C(C(=O)N2CCN(C)CC2C(=O)NC2(CO)CC2)SCCO1 68168,Cc1nc2c(N3CCN(C(c4c(F)cncc4F)=O)C4CC34)ncnc2[nH]1 68169,N(C1CCc2ccccc21)C(CCCCNC(=O)C=CC1CCOC1)=O 68170,c1(C(N2CCC(OCC(N3C(C)CC3CO)=O)C2)=O)cc(C#N)n(C)n1 68171,c1(C(N2C(CC(C)C)CCC2)=O)cccc(S(=O)(=O)NCc2cc(O)no2)c1 68172,c1(C(=O)OCC)nc(C(N2CCC(C(C)NC(=O)CC3CCC3)C2)=O)cs1 68173,c1(C(N(C2CCCN(C(C3(C(F)F)CCC3)=O)C2)C)=O)nn(C)nc1C(F)(F)F 68174,c1(N2C(C)CCC(NC(Cc3cc(COC)on3)=O)C2)nc(OC)c(F)c(C)n1 68175,N1(CCCC)CCN(C(c2c(C)cnn2COC)C(=O)NC)CC1 68176,Cc1ccc(C#N)c(NC(C2CC(NCc3cncs3)C2)=O)c1 68177,N1(C(C(=O)Nc2ccc(F)cc2)c2csnn2)CCc2ccc(Cl)nc2C1 68178,c1(OC)c(C)csc1C(N1CC(F)CC1CN(C)C(c1cnc(C)[nH]1)=O)=O 68179,c1(C(=O)NC(CC2CN(c3snc(COC)n3)C2)C)ncc(F)cc1F 68180,c1(NCCCC(=O)NC(C2(CC(=O)O)CC2)C)ccc(C#N)c([N+](=O)[O-])c1 68181,C1(NC(C(C=C)(C)O)=O)CCC2(CC1)CN(C(c1ccccc1C(=O)OC)=O)C2 68182,C1(CC)CCC(C)N(C(c2ccc(CNC(c3nc(C4CC4)cs3)=O)nc2)=O)C1 68183,CCC(C(=O)OC)C(=O)NC(C)(C)CN(C(=O)C(COC)OC)C 68184,c1(C(N2C(CN(C(=O)CSC)CC)CCCC2)=O)ccc(C(F)(F)F)c(F)c1C 68185,C(=O)(CC(CNC(C1CSCC(=O)N1)=O)C1CCC1)NCc1c(C)occ1 68186,C12(C(=O)NCC(CNC(Cc3nc(=N)[nH][nH]3)=O)F)CC3CC1(CO)CC3C2 68187,c1(C(=O)NC2CCC2CNC(c2cc(SC(F)(F)F)c[nH]2)=O)ncc(F)cn1 68188,N1(C(CCSCC)=O)CCC2CCN(C(=O)COCC3CCC3)CC12 68189,C12(C(N(CCNC(=O)CCSCC(C)C)CC)=O)CC(C)C1C2 68190,c12cnc(F)cc1C(=O)N2.N1(CC)CCC(NC(=O)CCNS(C)(=O)=O)C1 68191,C1(CC)CN(C(=O)CC2CCC(NC(=O)CCCC3CC3)C2)CC1F 68192,C1(O)(C(C(=O)NC2C(O)CC2O)NC(CC)=O)CCCCC1 68193,C(=O)(CCCC(F)(F)F)NC(C)CCCNC(c1cnc(-n2cccn2)cn1)=O 68194,CC(CCCNC(c1csc(O)n1)=O)NC(c1csc(O)n1)=O 68195,c1(C(=O)NCCC(=C)CNC(=O)CC2CCCOC2)ccccc1SC 68196,C1(C(=O)OC)(NC2CC(OC)C(N3CCOCC3)C2)CCC(F)(F)CC1 68197,C(CCC(C)CC(=O)N1CC2CC1CN2C(=O)C=C(C)C(C)(C)C)=C(C)C 68198,N1(C(C=CCCC)=O)CCC2(CCCC2NC(c2cnc(N(C)C)o2)=O)C1 68199,c1(CC(N2CC(C)C(CNC(c3cc(Br)c[nH]3)=O)C2)=O)nn(C)c2ccccc12 68200,C1(C(=O)NC2C(CNC(=O)CC3(O)CCC3)CC2)(NC(N)=O)CCCCC1 68201,C(=O)(C1c2c[nH]nc2CCC1C)NC1C(S(CC)=O)CCC1 68202,CN1CC(NCc2cccc([Si](C)(C)C)c2)Cc2ccccc21 68203,C(=O)(C(O)C(C)CC)NCC(CCC)NC(=O)COC1CCCCCC1 68204,n1(C(CC)C)nc(C(=O)NC(C)CNC(=O)C=Cc2csc(C)n2)cc1C 68205,C(=O)(C(F)C(C)CNC(=O)C(C)(C)C(F)F)NCCc1c(C)ncs1 68206,c1(CNC(C2CC2CNc2cncc(C(F)(F)F)n2)=O)csc2ccc(Br)cc12 68207,c1(NCc2cccc(C(=O)Nc3ccccc3CCO)c2)nc(Cl)c(Br)cc1O 68208,c1(N(C2CCCN(C(CCC(C)SC)=O)C2)C)snc(C)c1C#N 68209,C1(NC(C2CCOCC2)=O)CN(C(=O)Cc2cocc2Br)CC12CC2 68210,c1(C(=O)NC2C(F)CCN(C(C=Cc3c(C)ncs3)=O)C2)ccc2c(c1)CCC2 68211,c1(NC(C2(O)CCN(C(=O)Cc3cc(F)ccc3Cl)C2)=O)cccc2[nH]ccc12 68212,Cc1c(C(=O)NCC(C(=O)Nc2ccccc2C(C)(C)C)N(C)C)cccc1O 68213,C(N=c1[nH]c(=NC2CCCCCCC2)[nH]c2c1SCC2)C1N(CCC)CCCC1 68214,c1(C(N(C(C)C(=O)NCC2CCC2CO)CCC)=O)ncc2ccccn12 68215,C1(NC(c2c(C)onc2)=O)(CNC(c2cnoc2C2CC2)=O)CC2CCC1C2 68216,C1(CC(=O)NC)CN(C(=O)Cn2cnc(=N)[nH]2)CCN1C(=O)CC1CC1(Cl)Cl 68217,C1(C(=O)NCC2(CO)C(C)(C)C2)CCOCCN1C(c1ccc(C#N)o1)=O 68218,c1(C(=O)NCC2C(NC(C3(C)C=CCCC3)=O)CCC2)cc(F)c(F)c(O)c1F 68219,c1(C(=O)NCCN(C(C2CCC(=O)NC2)=O)CC)coc2ccccc12 68220,C=Cc1cc(C(=O)NCC2(C)CCN(C(c3ccnc(OC)c3)=O)C2)cc(F)c1 68221,c1(COC)nn(C)c(Cl)c1C(N1CCCC1CNC(C1CC(C)(C)C1)=O)=O 68222,Cc1ccc(C=CC(=O)NCC(C2CC2)NC(=O)C(n2nccc2C)C)cc1Cl 68223,C1(CC(=O)NCC(CC)C(C)C)CCN(C(=O)CCC2CCC(=O)C2)C1(C)C 68224,c1(CSc2nc(CCC(CCC)O)on2)cc(C(N)=O)cc2cccnc12 68225,N1(C(CSC)=O)Cc2ccccc2C(CNC(c2cnc(NC(C)=O)o2)=O)C1 68226,C1(CNC(C=C(C)C(C)(C)C)=O)CC2CN(C(C3(C#N)CC4CC4C3)=O)CC12 68227,CCC(CC(=O)N(CCC(=O)NC(C)(C)CC(C)C)C)CC(C)C 68228,N1(C(=O)Cn2cnc(Br)c2)CCC2CCCC(C1)N2C(C1C2COCC12)=O 68229,C1(C(=O)NC(C)C(C)(C)NC(=O)C=CCN2CCCC2)CS(=O)(=O)CCO1 68230,C1(NC(c2cn(C)c(=O)nc2O)=O)CC(C2CCN(C(=O)CC3CC3)C2)C1 68231,CC(C)(O)C(F)C(=O)N1CCOC(c2cn(Cc3cncc(N)c3)nn2)C1 68232,N1(C(c2ncn(CC)c2)=O)CCC(C2CCN(Cc3cc(C)ccc3C)C2)C1 68233,CC1(C)CN(C(c2ccon2)=O)CC1NC(c1cc(-c2ccco2)cs1)=O 68234,CCCCS(=O)(=O)NC(N(C)CCCc1cn(-c2ccccc2Cl)nn1)=O 68235,N1(C(CCCN(C)C)=O)CC2CC2C1C(=O)NC(C1CCOC1)CO 68236,C1(NC(C(CSC)O)=O)CCCN(C(c2cc3sccc3s2)=O)CC1 68237,CN1CCC(c2nnnn2CC2CC2)(NCC(=O)NCCC(O)C(C)(C)C)CC1 68238,C1(C2CCN(C)CC2)(C(N(CCCNC(C(C2CC2)OC)=O)C)=O)CC1 68239,CC1CCCC(OCCNC(=O)NCc2ccsc2)C1 68240,CC1(C(=O)NCc2cccc(Cl)c2F)CCCN(Cc2nccs2)C1 68241,c1(C(=O)NCC2CC(NC(CCN(CCC)C)=O)C2)ccc(OC)c(F)c1 68242,c1(OC)nc(C(=O)NCC2CCN(C(=O)CC3CCCC(C)C3)C2)sc1C 68243,c1(NC(C2N(Cc3ccc(OCC#C)cc3)CC(F)C2)=O)nc(Cl)cnc1Cl 68244,N1(C(c2cc(C)n(C)c2)=O)CC(N=[N+]=[N-])CC1C(=O)N(CC(O)CN(C)C)C 68245,N1(C(C)=O)CCCC(O)(CC(N2CC(O)(CNC(c3cc(OC)ns3)=O)C2)=O)C1 68246,CCC(CC)CC(=O)NCC1CN(C)CCN1C(=O)CCOc1ccc(Cl)cc1 68247,n1(CC)nccc1C(N1CCC(N(C(=O)COCc2ccnn2C)C)C1)=O 68248,CC1(CNC(=O)C2=CCCSC2)CCCN(C(=O)C(c2ccc(F)cc2)CO)C1 68249,C(=O)(CC(=O)NC1(CN(C)C(c2c[nH]nc2Cl)=O)CC1)NCC#C 68250,N1(C(C)=O)CCN(C(=O)CCCn2cc(CCOC(C)=O)nn2)CC1 68251,Cc1nn(C)c(C)c1C(N1CC(NC(=O)CCN2CCCS2(=O)=O)CC(O)C1)=O 68252,N=c1[nH]cc(C(=O)NCC(O)CNC(c2cscc2F)=O)c2cc[nH]c12 68253,C1(C(NOCC(O)C(C)C)=O)CCC(O)CN1C(c1cnncc1OC(F)F)=O 68254,N1(CC(N2CCN(C)CC2)C)CC2(CCC1CO)CC2 68255,c1(C(=O)NC2CCCN(C(C(CC)NC(C)=O)=O)CC2)cc(=O)c(OC)cn1C 68256,c1(C(=O)NCCC(C)(C)NC(C2C(OCC)C2)=O)snc(C)c1N 68257,c1(C(=O)NCCN(C(CCC2CC(OC)C2)=O)C)ccc(N)c2ccncc12 68258,C1(C2(O)CCOCC2)(C(N2C(C(=O)OCc3ccccc3)C(O)CC2)=O)CC1 68259,c1(OCC)cccc(C=CC(=O)N(C(C)CNC(=O)Cc2c(C)noc2C)C)c1 68260,c1(C(=O)OC)cccc(CCNC(=O)NC2CCC2C(C)(C)C)c1 68261,Cc1cnc(C(C)NC(=O)C(C2CCCCC2)C)s1 68262,C1(CCC)CN(C(=O)CCc2ncccn2)CCN1C(=O)CCCCNC(N)=O 68263,C(=O)(C(C)(CC)CO)N(CCC)CCc1nc(C(=O)NC)nc(O)c1 68264,CC1CCCN(C(c2coc(C3CCC3)n2)C(=O)NCc2ccccc2)C1 68265,C(=O)(C(O)C(C)(C)C)N1CC(C)C(NC(=O)Cc2ccncc2Cl)C1 68266,C#CCC(C)(CC)C(=O)N1CCCC(CC(N2CCc3sccc3C2)=O)C1 68267,C(c1ccc2occc2c1)=CC(=O)NCC1C(NC(C(C(C)O)C)=O)CCC1 68268,C(=O)(CC(C)CC(F)(F)F)N1C(CCCNC(C(=C(C)C2CC2)F)=O)CCC1 68269,CCC(CC)(CCO)NC(c1cncn1C(C)C)c1nnnn1C 68270,C1(C(=O)OC)COCC1C(=O)N(CCCCN(C(=O)C(C1CC1)NC(C)=O)C)C 68271,c1(NC(C(=O)NCCN(C(CC)C)C)=O)ccc2c(c1)C(=O)OC2(C)C 68272,C(CNC(=O)CCc1cnn(C)n1)(CCOC)NC(C(C)NC(CC)=O)=O 68273,c1(C(N2CCC(C(=O)OCC)CC2)=O)ccc(F)c(-c2c(C)cccc2F)n1 68274,C(=O)(C1=CCCSC1)NC(C(C)C)CNC(=O)COC1CCCOC1 68275,C1(NC(c2nc(CC)oc2C)=O)CN(C(C2CC2C(C)(C)C)=O)CC1N=[N+]=[N-] 68276,c1(C(=O)NC(CCCNC(C2C(=C)CC2)=O)C)cc(C)nn1-c1ccccc1 68277,N(C(=NCC1CCOc2ccccc21)NC1CCN(C(C)=O)CC1)C(C=C)C 68278,Cc1cc(C)n2nc(C(C)NCCOc3cccc(Br)c3)nc2n1 68279,c1(SCCCC)ccc(Cl)cc1C(=O)NCC(CC)NC(=O)C(F)CC1CCC1 68280,C12(NC(C(COC)COC)=O)CCC(F)(F)CC1CN(C(=O)C(F)C(C)(C)O)C2 68281,c1(C(=O)NC2CC(NC(c3nc(C)sc3C)=O)C2)ccc2nn[nH]c2c1O 68282,c1(C(=O)Nc2ccc(-c3cc(OC(C)C)ncc3)s2)cc(Br)cn2ccnc12 68283,C1(NC(C(C)C)=O)CCN(C(c2csc(C(C)(C)C)c2)=O)CC1CO 68284,C#CCCCCCC(=O)NCC1(F)CN(C(c2c(C)csc2C)=O)C1 68285,C12(CNC(C3N(C)CCC3)=O)CCCC(CN(C(=O)CC3CCC3)C1)C2 68286,O=S(=O)(c1cccc(-n2cnnn2)c1)NCC1=NOC2CCCC12 68287,c1(CNC(CCn2c(=O)sc(C)c2C)=O)c(F)ccc2c1OCO2 68288,C12(CNC(C=CCOC)=O)CC1CN(C(C1CC(C)CCO1)=O)C2 68289,C(=O)(CCCCCOCC)N1CCC(C(C(N2CCC(=C)C2)=O)C)C1 68290,c1(C(=O)NCCC(C(C)C)NC(=O)Cc2cn[nH]c2)cc(=O)c2ccccc2[nH]1 68291,C1(NC(C(C2CCC2)OC)=O)COCC1NC(c1ccoc1I)=O 68292,CC(Cc1ccccc1)(C(F)F)NC(=O)OCC(F)(F)F 68293,c1(C(=O)NC2CN(C(CC(C=C)C)=O)CC2O)n[nH]c2c1CS(=O)(=O)CC2 68294,c1(C(N2CCCC(CNC(CCC3CC(C)C3)=O)C2)=O)cn(C)c(=O)n(C)c1=O 68295,N1(C(C=C2CCC(C)CC2)=O)CCC(O)(C(C)NC(=O)CC(C)(F)F)CC1 68296,c1(CC)cc(C(c2nnnn2C2COC2)NC(C)CCC(C)C)ccc1C#N 68297,C#CC1CCC(NC(=O)COc2ccccc2F)CC1 68298,CC(C)(C)C(CNC(c1ccn(CCF)n1)=O)C(=O)NCC1(C)CC1(F)F 68299,C1(C(N(C)CC2CC2)=O)CN(Cc2cncn2C2CCCC2)CCC1O 68300,c1(C(=O)NCC=CCNC(=O)CC2(O)CCOCC2)cnn2c(=O)cc[nH]c12 68301,C1(CNC(C2(C)CC(C)C2)=O)CC2(CCN(C(=O)CNc3ccccn3)C2)CO1 68302,Cc1[nH]c(C)c(C(=O)NCC2=CCN(C(=O)C(C)Cc3cnc[nH]3)CC2)c1C 68303,C1(CNC(C(C)CN(C)C)=O)CCC2(CCC2)CN1C(c1cncn(C)c1=O)=O 68304,C1(CCNC(CCOCCCOC)=O)CN(C(=O)CC2CS(=O)(=O)C2)CCO1 68305,c1(OC)cc(C(=O)NC2CC(C)CN(C(=O)OC(C)(C)C)C2)ccc1C 68306,N1(C(C(CCOC)OC)=O)Cc2ccccc2CC1CNC(=O)CC1CCCC1 68307,c1(CC(=O)NCCC(Cn2cc(C=CC)nn2)(F)F)ccc(C#N)cc1F 68308,Cc1nocc1CCC(=O)NC1CC(CNC(c2csnc2Br)=O)C1 68309,C1(C(=O)NCCc2ccc(O)cn2)CCc2nnc(-c3ccccc3)n2C1 68310,c1(CC)oc(C(=O)NCC2CN(C(=O)C(CC3CC3)CC3CC3)CC2C)cc1C 68311,C1(COC)(CNC(=O)CCc2cc(C)no2)CCCN1C(C1CCCC1)=O 68312,c1(CCC(=O)NCC(CNC(c2cc(CC)on2)=O)(C)O)c(C)n[nH]c1C 68313,C1(CC(=O)NC(CSc2nc[nH]n2)CO)CC2(C1)CN(C(=O)CC1CC1)C2 68314,N1(C(c2c(C)nncc2)=O)CCN(C(c2ocnc2C)=O)CC(O)C1 68315,c1(N(C)C)nccc2c1CCN(Cc1ncsc1Br)C2 68316,C(C)(C)(CCCNC(C1CCC(C)O1)=O)NC(c1c(C(C)C)ncs1)=O 68317,C1(CCNC(C(C=CCCC)O)=O)CCCN(C(=O)CNC(=O)CCC(C)C)C1 68318,N1(C(C(C)(O)C2CCC2)=O)CC(NC(C2CC3(CCOC3)C2)=O)CC2(CCC2)C1 68319,C1(NC(C=C(C)C(C)C)=O)CCN(C(C23CC(C)(CCO2)C3)=O)CC1CO 68320,Cc1cc(C(Cc2cn(C3CCOC3)nn2)NCc2ccco2)on1 68321,c1(N(C(C)CN(C)C)C(C2COC3(CCNCC3)C2)=O)ncc2cccc(Br)c2n1 68322,C1(C)(C(N(CC(=O)NCC)C)=O)CC12CCN(C(c1cccc(SC)c1)=O)CC2 68323,c1(C(N(C(CNC(C(C)CC2CCC2)=O)C)C)=O)c[nH]c2nccc-2c1 68324,C1(CNC(c2ccn(CC)n2)=O)CC(NC(=O)C(O)Cc2cnn(C)c2)C(O)C1 68325,N1(C(CCOCC)=O)CCN(C(C23CC(C2)S(=O)(=O)C3)=O)CC1C 68326,c1(C(N(C2CCN(C(=O)C3=NNC(=O)CC3)C2)C)=O)cc(F)c2cn[nH]c2c1 68327,Cc1nc(CC(=O)NC2(C(=O)N(C)C(C)C3CC3)CSC2)cs1 68328,N1(C(C2(CC(C)C)CCNC2)=O)CCC(C#N)(NC(N)=O)C1 68329,c1(C(N2C(CN(C(CC3N(CC)CCC3)=O)C)CCCC2)=O)cc(N)nc(Cl)c1 68330,N1(C(CNC(CCC(C)C)=O)=O)CCC(C(=O)N(C)Cc2ccsc2)C(C)(C)C1 68331,CC1(CO)CCCN(C(C2CCC(O)CN2C(C2CCS(=O)CC2)=O)=O)C1 68332,c1(COC)cnc(OC)c(C(=O)NC2CCC2NC(=O)CN(C)C2CC2)c1 68333,C(=O)(C1=C(Cl)CCCC1)NC1(O)CCN(C(CCOC(CC(C)C)C)=O)CC1 68334,CCC(CC)C(C)C(=O)NCC1CC(NC(C2(CN3CCCC3)CC2)=O)C1 68335,c1(CN(C(CN(C)CC)=O)C)ccc(CC2(C(=O)NC)CC2)cc1 68336,N1(C(c2scc(C)c2Cl)=O)CCC(CNC(=O)CCC2CCC(C)O2)C(F)(F)C1 68337,c1(C(N2CC(c3cn(C4(C(=O)OC)CC4)nn3)(C)C2)=O)ccnnc1C 68338,C(=O)(C1CCc2ccccc21)NCc1c(C(=O)NC2(CCC)CCC2)con1 68339,N1(C(c2cnc(CC(C)C)s2)=O)CC2CC(NC(=O)CC3=NNC(=O)C3)CC1C2 68340,CCCC(C)(CC)C(=O)N1CCCCCC(NC(C2(O)CCC2)=O)C1 68341,O=C(C1=COCC1)NCC1CN(C(=O)Cc2cccc(OC3CC3)c2)CCO1 68342,C1(CC(=O)N(CC(C)NC(=O)C(c2ccccc2)C)C)(CC)CCOCC1 68343,C1(OC)CCC(C(=O)NC2(CCC(=O)NCc3ccc(C)cc3)CCCC2)CC1 68344,C12(CNC(C(C(C)(C)C)SC)=O)CN(C(=O)C(F)=C(C)C3CC3)CC(F)(C1)C2 68345,Cc1nc(N2CCC3(CCN(C(=O)C(C)n4ccnc4)C3)C2)c2sccc2n1 68346,c1(C(=O)OC)cccnc1C(=O)N(C)CCOCCN(C(=O)C(F)C1CCC1)C 68347,CC1=NS(=O)(=O)N(C)C=C1C(=O)NCCC(C(C)C)NC(=O)C=CC(=O)N(C)C 68348,C1(C(N2CCC(C)(NC(c3nc(C(C)(C)C)oc3)=O)C2)=O)CC12CC(F)(F)C2 68349,N1(Cc2cn(C(C)C)nc2)C(C(N2CCC(n3cnnc3)CC2)=O)CC2CC12 68350,C1(C(=O)Nc2ccc(CO)cn2)CN(C(C2(C3CC3)CC2)=O)CC1C1CC1 68351,C(=O)(C(O)CCC(F)(F)F)NC(C1CCCC1)CNC(CC(COC)(C)C)=O 68352,c1(C(N2CC(NC(Cc3c(C)cccn3)=O)C(C)C2)=O)c(C)nc2cccnn12 68353,C1(CNC(=O)Cc2ccc(Cl)s2)C2CN(C(=O)CCc3cncc(F)c3)CC12 68354,N1(C(=O)COc2ccsc2Cl)CCC(O)C(O)c2ccccc21 68355,c1(C(N2CCC(C(N3CCCC(C(=O)OC)C3)=O)C2)=O)c(F)ccc(Br)c1OC 68356,Cc1ccc(C=CC(N2CCN(C(=O)Cn3ccnc3C)C(C)C2C)=O)cc1Cl 68357,C1(NC(C(CCC)O)=O)CCCN(C(C2CC3(CC(OC)C3)C2)=O)C1C 68358,CCCCC(CC)CC(=O)N1CC(F)CC1CN(C(=O)CC(C)(C)C(F)F)C 68359,C1(NC(C2C(C)CN(C(c3cnc(O)o3)=O)C2)=O)CCN(C)CC1C#N 68360,C(CC(C(=O)NCCCOCCNC(=O)C=Cc1ccoc1)NC=O)SC 68361,C(=O)(CC1=NNC(=O)C1)N1C2C(NC(CN(C)C(N)=O)=O)C(C2)C1 68362,O=C(C#CC1CCOC1)NCC1CCN(C(=O)CCOC2CCCC2)CC1O 68363,C=CC1CCCC(c2nnnn2CC2CC2(Cl)Cl)(NCc2ccc(C3CC3)o2)C1 68364,C(CC(=O)NCC(C)(C)N1CCCC1)(C(F)F)NC(C(COC(C)C)(C)C)=O 68365,C1(c2n(CC(=C)C)nnn2)(NCc2ccccc2-n2cncn2)CC(C)N(C)C1 68366,c1(C(=O)NCC(C(=O)NCC(COCC)C)O)ccc2[nH]ccc2c1 68367,Cc1csc(C(=O)NC(CNC(c2cnccc2C(F)F)=O)C2CC2)c1Cl 68368,c1(NC(C(C2CCC2)NC(c2c(CC)cco2)=O)=O)ccc(O)c(OC)c1 68369,C1(CNC(CN2CCC(C)CC2)=O)CN(C(=O)Cc2cn(C)nn2)C(C)(C)C1 68370,c1(NC(=O)NCC2(NC(C3CN(S(C)(=O)=O)C3)=O)CCOC2)c(C)ncn1C 68371,C(=O)(C(C(=O)NCC12CC1CN(C(C1CCC1COC)=O)C2)C(C)C)OCC 68372,c1(C(=O)NCC2(C)CCN(C(C(C(C)C)NS(N)(=O)=O)=O)C2)cccc(=O)n1O 68373,C1(CC)COCCN(C(C2CCCN(C(c3cnn(CC)c3C)=O)C2)=O)C1 68374,c1(C(=O)NC2CCCCN(C(C(C(C)C)(C)C)=O)C2)cc2c(nc1N)CCC2 68375,c1(C(=O)NCC2N(C(C(C)Oc3cccnc3)=O)CC2)cnccc1C1OCCO1 68376,N1(C(C)C)CC(C(N2CC=CC(NC(=O)C(=O)NCC(F)(F)F)C2)=O)CC1=O 68377,C1(C(=O)NCc2c(C(=O)NCC(C3CC3)SC)con2)CCC(C)=C(C)C1 68378,C1(C(COC(n2cccc2N(C)C)=O)=O)CCCN(C(=O)C(C)(C)C)C1 68379,C(C(O)C(=O)NCC1CC(C(=O)N(C2CC(F)(F)C2)C)C1)SC 68380,C1(C(=O)NCC2(C(C)(C)O)CN(C(=O)CC(O)C3CCCC3)C2)CC12CCCCC2 68381,C(=O)(C(C)(C)CS(N)(=O)=O)N(CCC1N(C(CCC(=O)N(C)C)=O)CCCC1)C 68382,C(=O)(CC1=CCN(C(C2OCCC2(C)C)=O)CC1)N(C(CSC)C)C 68383,Cc1cccc2nc(C(=O)NCC(O)CNC(C34CCCCC3C4)=O)cn12 68384,C1(F)(CNC(C2C(OC(C)=O)C2)=O)CC(CNC(C2(F)CC2)=O)C1 68385,c1(C(=O)NCCC(=C)CNC(=O)C(c2ccnn2C)C)cc(F)cc(F)c1 68386,c1(CC)ncc(C(N2CCC(CC(N3CCNC(=O)C3CC)=O)C2)=O)c(C)n1 68387,CC1CCN(Cc2cccc(-c3cc(C(=O)NN4CCCC4)n(C)n3)c2)CC1C 68388,c1(CC)nn(C)c(C(=O)NC2CCN(C(=O)C(C)(C)Cl)C2)c1Cl 68389,N1(C(=O)OC)CCN(C(C2CCCN2C(=O)C=Cc2ccsc2)=O)CC1 68390,CCC(C)C(CC(=O)N1CCn2nncc2C1)NC(=O)CSCC(F)F 68391,c1(OCCCC(=O)NC2C(COC)COCC2)ccc(F)c(F)c1 68392,C(=O)(CCCCNC(N)=O)NCC(C)(C)CNC(C1(C)CCNC1=O)=O 68393,C1(NC(CCC=C=C)=O)CCN(C(=O)CCC2CCOC2)C12CC2 68394,C=CC(C)CC(=O)NC(CNC(=O)CC1CNC(=O)O1)C(C)C 68395,C1(CC(=O)NC2CCC(CNC(CCC)=O)C2)CC(=O)NC(=O)C1 68396,N1(C(C2N(C)CCC2)=O)CCCC(NC(C2CC(F)C(=O)N2)=O)C1 68397,Cc1ccc(-n2nnnc2N2CCC(COC(C(=O)C#CC3CC3)=O)CC2)cc1 68398,c1(N2CCC(F)(CNC(c3ccc4nccn4c3)=O)C2)ncnc2[nH]cnc12 68399,c1(C(=O)NC(CNC(C(CC)c2cccnc2)=O)CO)ccc(Cl)nc1O 68400,c1(N(C)C)ccc(CN2C3CN(Cc4ccnc(OC5CCC5)c4)CC32)c(O)c1 68401,C1(C(=O)NC2(CO)CN(C(C(=Cc3cnc[nH]3)C)=O)C2)CCS(=O)(=O)N1 68402,c1(C(=O)NCCC2CC(NC(Cn3cc(C(C)=O)nn3)=O)C2)ccc(F)cn1 68403,CCC(F)(C(=O)OC)C(=O)NCCNC(c1ccc(CCF)cc1)=O 68404,N1(C(C(C)CCN(C)C)=O)CCC(C2CC2)C1CNC(=O)C=CC1CC1 68405,Cc1noc(C)c1C(C)C(=O)NCCCNC(c1ccc(NS(C)(=O)=O)nc1)=O 68406,C12(CC)CCC(C(=O)NCCCN(C(C3CCCC(=O)O3)=O)C3CC3)(CC1)CO2 68407,CN1CC(C)(C(N2CC=CC(C(=O)NCC(N3CC=CC3)=O)C2)=O)CC1=O 68408,C1(CN2CC(c3nc(C(C)C)[nH]n3)OCC2)CCCCCCC1O 68409,c1(CNC(CC(C)CC2CCC2)=O)ccccc1[N+](=O)[O-] 68410,C1(C(N2CCC(CC(F)(F)F)CC2)=O)COC2(CNC2)C1 68411,C12(CC(=O)NC3(Nc4ncc(F)cn4)CCC3)CC3CC(CC(C3)C1)C2 68412,N1(C(C2CC=C(C)CC2)=O)CCC(C)(C(=O)Nc2ncc(C)c(Cl)n2)CC1 68413,CN1CCCC1(C)C(=O)NCC1CCN1C(=O)Cn1[nH]cnc1=N 68414,C(N=c1[nH]cnc(Cl)c1C(C)=O)C1CCC(NC(C2(COC)CCOC2)=O)C1 68415,n1(C(C(=O)NCC(CC)NC(=O)CCn2ccnc2)C)nc(C)cc1C 68416,N1(C(CCCC#C)=O)CCCC2C(NC(c3cc(O)cc(C#N)c3)=O)C(C)(C)C12 68417,C=CCCC(=O)N(CCCCCNC(=O)C=CC(=O)NC1CC1)C 68418,c1(SCC(=O)NCC(C)NC(C(C)NS(CCC)(=O)=O)=O)nc2ccccc2s1 68419,c1(C(N(CCC)CCNC(C2(C(N)=O)CCC2)=O)=O)cc(Cl)cc(Cl)n1 68420,c1(CC(=O)NC2CN(C(c3c(OC)nsc3)=O)C3C2C3)cc2ccccc2o1 68421,c1(C(=O)NC2COCCN(C(C3CC(C(C)C)C3)=O)C2)cn2ccccc2n1 68422,N1(CC=CC(=O)NC2(c3cccs3)C(C)(C)C2)CC2C(CNC(=O)C(N)=O)C2C1 68423,C(=O)(C(C(C)(C)C)NC(N)=O)NCCC(C)N(C(=O)C(=O)Cc1ccccc1)C 68424,c1(C(N2CC(O)CC(NC(C3SCCS3)=O)C2)=O)cnn2c(Cl)cccc12 68425,C(=O)(C#CC1CCCC1)NC(C1(O)CCN(C(CCCOC(C(C)C)=O)=O)C1)C 68426,CCC(C)C(CC(=O)N(CC(F)F)CC)NC(C1CCC2(CCC2)C1)=O 68427,c1(C(=O)NCCC2CN(C(C3C(C(=O)OC)CCC3)=O)C2)c(C)cccc1O 68428,C1(C(N(CC(=O)NCCC2(F)CC2)C)=O)CCCN1C1CC1 68429,C(C(=O)NC1CCC1)(C1=Cc2cc(Br)ccc2OC1)N(C(C=C)C1CC1)C 68430,Cc1c(C)n(C)c2ccc(C(=O)NCC3CN(C(=O)CO)CCC3C)cc12 68431,C1CC2(CCNCC2)C1.c1(C(C(=O)N(CCC#N)C)N)cccnc1 68432,N1(C(CCOCC)=O)C2CCCC1CN(C(=O)C(c1ccccc1)=O)C2 68433,Cc1cncc(CCC(=O)NC2CC(C)N(C(=O)CCOC(C)C)C2)c1 68434,C(=O)(CCC(CC)NC(=O)CCCCOC)N1C(C=C)CCC1 68435,C1(C(N2CCC(C(C(=O)OC)(C)C)C2)=O)CC(=O)N(C(C)(C)C)C1 68436,C1(NC(Cn2nc(C)c(Br)c2)=O)CN(C(c2cnc(N)cn2)=O)CC1(C)C 68437,CCC(C(=O)NCC(C)(C)NC(C1CC1c1cncn1C)=O)SC 68438,C1(NC(C2CC3(CCC3O)C2)=O)CCC(O)CN(C(c2cc(CO)on2)=O)C1 68439,Cc1ccc(F)cc1CN1CC(NC(c2cnc(C)c(C(F)(F)F)c2)=O)C(O)C1 68440,c1(C(N2C(CN(C(COC(CC)C)=O)C)CCCC2)=O)ccnc2ncsc12 68441,C(=O)(CN=c1[nH]cncc1I)N1CCC(Nc2c(C(N)=O)cccn2)CC1 68442,C1(NC(CCCC)=O)CCC2(CC1)CC2NC(C1CCC(=O)N1C)=O 68443,C(=O)(CC(C)(C)NC(=O)Cc1ccccn1)NC(C(=O)OCC)C 68444,C#CC1CN(C(=O)CC2CC(F)CN2C(=O)CC2CNC(=O)O2)CCN1C 68445,C1(NC(c2c(C(C)C)noc2)=O)CN(C(C2COC(=O)N2C)=O)CC1O 68446,CCCCC(=O)C(=O)NC1CCC1C(N1CC(C2CC2)OC(C)C1)=O 68447,N1(CCC(=C)C)CCC2(CCCN(C(C3(c4cccnc4)CC3)=O)C2)C1 68448,C(=O)(CS(=O)(=O)CCC)N1CCC(C(N(C2CC3(CCC3)C2)CCCC)=O)CC1 68449,C1(O)(CCNC(Cc2ccc(C)nc2)=O)CCN(C(=O)C(C)(C)CC#N)CC1 68450,N1(C(c2cc(Cl)c(Br)c(Cl)c2)=O)CCC2C(CCN2C(c2cc[n+]([O-])cc2)=O)C1 68451,C1(C(=O)NC2C3CN(C(CC(CC)CC)=O)C2CC3)CCc2nnnn2CC1 68452,Cc1nn(CC(=O)NC(C)(CO)C(=O)NCCC(O)C(C)C)c(=O)o1 68453,n1(CC)nnc(-c2nc(CC(C)CC)nn2-c2ccc(OC(C)(C)C)cc2)c1C 68454,C=CCC(C)C(=O)NC(c1ccc(CNC(=O)CCc2cnn(C)n2)cc1)C 68455,c1(C(=O)NCC2CC(NC(=O)C=Cc3ccccc3)CC2O)cn2c(n1)CCC2 68456,C1(C(N(CCNC(C(CC)Oc2ccccc2C)=O)C)=O)C2CCC1(C)C2(C)C 68457,C1(C(N(CCC(C)NC(c2cc(C3CC3)ccc2F)=O)C)=O)CCC(C)(C)CO1 68458,C1(C(=O)OCc2cn(C)nn2)CC2CC(O)C(O)C(C1)C2 68459,Cc1cnc(C(=O)NCc2ccc(C(=O)NC3CC(C4CC4)C3)nc2)cn1 68460,Cc1cncc(C(N2CCCC2CCCNC(=O)C(C)OCC2CC2)=O)c1C 68461,Cc1ccc(Cl)cc1NC(=O)C(C)(C)C1CCCN1C(=O)CC(C)N(C)C 68462,c1(CCCC(=O)N(CCNC(C=CC=CC)=O)CC)cccc(Cl)n1 68463,c1(CC(=O)NCC=CCNC(C2C(COC)C2)=O)ccc(F)c(Cl)c1 68464,N1(C(C(CCC)CNC(=O)CN2CC(C)(C)C2)=O)CCC2(CCCOC2)C1 68465,Cc1nc(NCCS(C)=O)cc(N2CCCC(C(F)(F)F)C2)n1 68466,c1(OC)ccc(C)c(NC(=O)CC2CN(C(=O)CCC3CCCN3C)CCO2)c1 68467,c1(C(N2CCC(NC(COCC#C)=O)CC2C)=O)cc2nc[nH]c2cc1F 68468,C(=O)(C(C)(F)C(=O)N1CC=CC(C(=O)N(C)CCc2ccccn2)C1)OC 68469,C1(OC)CC(C)(C)C(=O)N1CN1CCC1CCO 68470,N1(C(CNC(=O)OC)=O)CCCC2CN(C(=O)CC3CCCCC3F)CC12 68471,C1(C(=O)NCC2(Cl)CC2(F)F)COC2(C1)CN(C(=O)CCSC1CCC1)C2 68472,c1(C(=O)NC2(COC)CC(OC)C2)csc(N=S(C)(C)=O)n1 68473,C#Cc1ccc(C(N2CCC3(CC(NC(=O)CCCCSC)C3)C2)=O)cc1C 68474,CCCCCCCCC(=O)NC1CCC(NC(c2csc3ccccc23)=O)CC1 68475,N1(C(c2cccc(C(C)=O)c2)=O)CCCC(O)(CN(C(=O)C(C)NC(N)=O)C)C1 68476,c1(N(C)C)ncc2c(n1)CN(c1cc(NC(=O)NCCCl)ncn1)C2 68477,c1(C(=O)NC(C2CCN(C(C3=C(C)OCC3)=O)C2)C)cc(C)cc(Cl)c1N 68478,C1(C(C)C)CC(NC(C2CC(C)N2C(=O)C(C)(C)Cl)=O)CO1 68479,Cc1cccnc1CC(=O)NC(CN(C)C(C1CCC(CO)CC1)=O)(CO)CO 68480,c1(-c2c(OC)ccc(-c3nccn3CC(O)CO)c2)cc2cccc(OC)c2o1 68481,C(CC(C(=O)N1CC(C(=O)NCC2(F)CCCCC2)(SC)C1)OC)OC 68482,c1(C(CNC(c2ccc(C3CC3)o2)=O)NC(=O)C2CC2)ccccc1Br 68483,N1(C(c2c(N(C)C)nccc2)=O)CCN(C(=O)C=CCF)CC1C1CCC1 68484,C(CCCCCCC(=O)NCCOCCN(C)C(C1CC2CCC1O2)=O)SC 68485,C1(NC(C2N(C(c3c(C)n(C)nc3)=O)CC=C2)=O)CC2(CNC(=O)O2)C1 68486,C1(NC(=O)CCc2cncs2)C=CCC(C(=O)NCCCCn2ccnc2)C1 68487,Cc1ccc2cc(C(c3nnnn3C(C)C)NC3COC4(COC4)C3)n(C)c2c1 68488,n1(CCNCC(C)(C(C)C)N(CC)Cc2cccnc2)nc(C)c(C)c1C 68489,C1(CC)CN(C(=O)C(c2c(C)n[nH]c2C)C)CC1NC(=O)C(C)NC(C)=O 68490,N1(C(CCCCCOC)=O)CC2CCOC2(CNC(=O)Cc2nc(C)sc2C)C1 68491,c1(OCC)ccc(C(=O)NC(C)C(C)NC(=O)C2=C(C)CCC2)cc1OC 68492,c1(CC(=O)NC2CC(CNC(Cc3c(C)ncs3)=O)C2)sc(O)nc1O 68493,N1(C(C(CC)CC)=O)CCCC(C)(C)C1CNC(c1c(C)ncnc1C)=O 68494,c1(COC(N(C)C)=O)ccc(NC(=O)CC(c2ccccn2)N(C)C)cc1 68495,CC(CC(C)(F)F)C(=O)NC(c1cn(CCN2CCNC2=O)nn1)(C)C 68496,Cc1cnncc1C(=O)NC(CC1CC1)CC(=O)N1CCN(c2cccnn2)CC1 68497,C1(C(N(C2CCN(C(=O)Cc3sccc3C)C2)CC)=O)Cc2nccnc2C1 68498,c1(C(C)=O)cc(Cl)c(N(C)C(c2ccccc2N2CCCC2)=O)nc1C 68499,c1(OCC(=C)C)cc(CN(C)C)ccc1OC.O1NC(=O)NCCC1 68500,c1(C(C(=O)NCC(CCOC)NC(c2sccc2C)=O)(F)F)ccc(C)cc1 68501,N1(C(C2=C(C)OCCC2)=O)CCOC2(C1)CN(C(=O)CC13COC(CF)(C1)C3)C2 68502,c1(NC(N(C(C2CCCCC2)C)C)=O)ncc(Br)cc1Cl 68503,c1(OC)cc(OC)c(F)c(C(=O)NC2CC(F)CN(C(C3CCCS3)=O)C2)c1 68504,c1(C(=O)NCC(C2CCOC2)NC(=O)C=Cc2cccs2)cnnc(C2CC2)c1 68505,Cc1nc2ncnn2cc1C(=O)NC1CCCCC1NC(=O)Cc1cccnc1 68506,C1(NC(CN2CC(=O)NCC2)=O)CCCC12CCN(C(=O)Cc1cccs1)CC2 68507,c1(CNC(N(C)Cc2cc(F)cc(Br)c2)=O)ccc(S(N)(=O)=O)cc1Cl 68508,C1(CC)(NC(=O)C(C)C(C)(F)F)CCN(C(=O)C(C)Cc2ccncc2)CC1 68509,C1(CNC(c2ccc3[nH]ccc3n2)=O)CCCC2CN(C(=O)C3CC3)CC12 68510,C1(CC(=O)NC2(c3ccccc3)CCCC2)CN(Cc2cc(Br)cs2)CCO1 68511,C(C(O)C(=O)NC1(C)CC(NC(c2cc(C3CCC3)[nH]n2)=O)C1)=CC 68512,c1(N(C)C)cncc(C(=O)NC2CC(CO)N(C(=O)C(N3CCOCC3)C)C2)c1 68513,CC1CCc2nc(N3CC4CSCC(C4)C3)[nH]c(=NCC(Cl)(Cl)Cl)c2C1 68514,c1(C(=O)NC2C(C(N(CCCC(O)CO)C)=O)COCC2)ccc([N+](=O)[O-])[nH]1 68515,c1(C(=O)NC(C(=O)NC(CC)C(=O)NC)CC2CCC2)ccn(C)c(=O)c1 68516,CC(C)C(CC(=O)NCC1CC2CCC1CC2)NC(C1CC2(CCO1)CC2)=O 68517,c1(C(N2CC(C)(CNC(CCCCOCC)=O)OCC2)=O)c(F)ccc(O)c1F 68518,C1(CC)CN(C(c2cc(-c3cccnc3)no2)=O)CCN1C(=O)C1=CCC1 68519,C(=O)(C1=C(Cl)CCCC1)NCCCC(C)NC(c1cc(CC)c(C)cc1)=O 68520,C(=O)(C(CN(C)C)CC)NCCCOCCNC(C(C)OCCCC)=O 68521,c1(C(CCNC(=O)NCC=CC)C)ccc(C(F)(F)F)cc1 68522,C(CC(C)CC)(C(=O)NCCC(=O)NCC)NC(CCCC)=O 68523,c1(C(C)=O)nc(SCC(=O)NCC(O)CN(C(=O)C(N2CCOCC2)O)C)cs1 68524,N1(C(C2(CNC(c3c(C)scn3)=O)CC3(CC3)C2)=O)CC2CC(C)C2C1 68525,C(=O)(CCCC(=O)NC1CCOC(c2cnn(C)c2)C1)c1ccc(OC)cc1 68526,c1(NC(C)=O)ccccc1CC(C)=CC(=O)NC1CC1NC(c1nocc1C)=O 68527,C(C1=NOC2CN(C(=O)Cc3cccs3)CC12)NC(C=Cc1cc(OC)ns1)=O 68528,C1(N(C)S(N)(=O)=O)(CO)CCN(C(C2CC23CC(F)(F)C3)=O)CC1.C(=O)CNC=O 68529,C(C(C)(C)C(=O)OC)(c1n(C(CC)(C)C)nnn1)NCC1(c2ccccc2)CC1 68530,c1(C(N2CCC(C)(CC(=O)NC(CCO)C3CC3)C2)=O)cc2ncccc2[nH]1 68531,C1(NC(C(C)(C)NC(=O)OC)=O)C2CCC(C2)C1C(=O)NCc1cncnc1 68532,c1(C(=O)NC2CC(CCNC(C3(Cl)C(C)(C)C3)=O)C2)cc2cn[nH]c2cn1 68533,c1(C(=O)NC2C(CNC(c3c(C)cns3)=O)COC2)cc(CC2CC2)ncn1 68534,c1(CNC(C2(CC)CCN(C(c3oc(CC)c(C)c3)=O)C2)=O)ccc(C)nc1O 68535,C1(C)(NC(C(C2CCCCC2)NC(c2c(C)snc2)=O)=O)CCC2(CC1)CC2 68536,C1(C(=O)NC2CCC(NC(CCC)=O)C2)COCCN1C1CCCC1 68537,C1(CN(C(=O)C2=CCSC2)C)CN(C(=O)C(C)(C)C2CCC2)CC12CC2 68538,C=C1CC2CC1CN2C(=O)C(C1(O)CN(C(=O)CC2CCC2)C1)F 68539,c1(C2C(C(=O)NCC(CNC(c3cccc(N)c3)=O)OC)C2)cccc(F)c1 68540,C(CC(=O)N1CCCC1)N(C(=O)COC(CSC)Br)C(C)C.C1C(=O)O1 68541,C(c1cnc[nH]1)=CC(=O)NCC(CN(C(=O)Cc1ccno1)C)O 68542,N1(C(CC2(C)CCN(C(C(C(C)(C)C)OC)=O)C2)=O)CC2(CCNC2=O)C1 68543,c1(C(=O)NCC(CC)NC(C2CCCCC2C(N)=O)=O)ccnc(OC)n1 68544,N1(C(C2(CCNC(=O)CC3CCCOC3)CC2)=O)CC2CCCC1C2CO 68545,N(C1CCc2cccnc21)C(CC1(C)CCN1C(=O)C1CC1)=O 68546,N1(C(C2(CC#C)CCCO2)=O)CC(CNC(c2cc(C)ncn2)=O)C(O)C1 68547,Cc1nc2n(c1CNC(c1c(C)sc3ccccc13)=O)CCCC2 68548,c1(C(=O)NC2CN(C(c3nn(C)c(Cl)c3)=O)CC2F)cccc2c1CCCO2 68549,Cc1nnc(C2CN(C(=O)NCC3CCC(O)C3)C2)o1 68550,N1(C(C2C(Cl)(C(=O)OC)C2)=O)CC2CCC(CNC(C3CC(C(C)C)C3)=O)(C2)C1 68551,C(=O)(C(CC(F)F)NC(=O)Cn1cccnc1=O)NC(c1ncccc1F)C 68552,C1(NC(c2ccc(-c3ccccc3)s2)=O)CCCN(C(c2ccncc2)=O)C1 68553,C1(c2nc(C(N3CCC(C)CC3)C)on2)COc2ccccc2C1 68554,N1(C(C(CC2CC2)NC(C2CC(F)(F)C2)=O)=O)CC2COCC2C1 68555,N#CC1(C(N2CC3(CCC3NC(=O)CCCc3ccncc3)C2)=O)CCOCC1 68556,C=C(C)CCC(=O)N1CCC(N(C(=O)C(=Cc2cnc[nH]2)C)C)CC1 68557,C#CC1(C(=O)NC2CN(CCC)C2)CN(C(=O)CCC=C(C)C)C1 68558,C1(F)(CNC(C(C)NC(C)(C)C)=O)CCN(C(=O)CC2OCCCC2(C)C)CC1 68559,N1(C(NN(C(C(C)NC2CC2)=O)C)=O)C(=O)Cc2ccccc2C1=O 68560,N1(CC(=O)Nc2scc(CC(=O)NC3(C(C)C)CC3)n2)CCN(C)CC1 68561,C1(C(C)NC(=O)N(CCO)CCO)CCCC(C(F)(F)F)C1 68562,c1(N2CCC(=CC(=O)Nc3c(C)ccc(O)c3)CC2)ncc2c(n1)NC(=O)C2 68563,c1(C(=O)NC2C(CNC(COC(C)=O)=O)COC2)cccc2c1CC(C)(C)C2 68564,Cc1ccc(Cl)c(OC(C)C(=O)NC2CN(C(=O)C3=NOC(C)C3)C2)c1 68565,C1(c2cn(C)nc2)CN(C(C2CC23CCCCC3)=O)CCN1C(=O)CCC(F)(F)F 68566,C1(C(N2CC(C)C(NC(C3(F)CCC3)=O)C2)=O)Cc2ccccc2S1(=O)=O 68567,N1(C(C(=O)NC2CCN(c3ccc(F)cc3F)C2)=O)CC2CCCCCC2C1 68568,C1(NC(C(C)CC2CCC2)=O)CCCC12CN(C(c1sc(F)cc1Cl)=O)C2 68569,C(=O)(CC(C(=O)NCCC1CCN(C(C2(N(C)C)CCC2)=O)C1)NC(C)=O)OC 68570,c1(OC)cncc(NC(C2CCC2NC(c2ccccc2C)=O)=O)c1 68571,Cc1cc2[nH]c(C(N3CC4=C(C3)CN(C(C3(C)CCCCO3)=O)C4)=O)cc2s1 68572,c1(C(N(CC(C)CNC(=O)CC2COC(=O)N2)C)=O)ncc(Cl)nc1Cl 68573,Cc1cccc2c1CC(C(N1CC3CN(C(=O)C(C)C(F)F)CC3C1)=O)O2 68574,CCCC(O)C(CO)NC(=O)CC1(N(C)C(c2[nH]cc(C)c2C)=O)CC1 68575,C(=O)(C1=NNC(=O)CC1)NC(C)CC(C)NC(c1cnc2n1CCS2)=O 68576,N1(C(=O)CCC2CCOC2)CCCCC(C(=O)NC2(C3CC3)CCCC2)C1 68577,N1(C(C2(CC)CC2)=O)C2CCC1C(C(=O)NCc1ncn(C3CC3)n1)C2 68578,c1(C(=O)NC23CCC(CN(C(c4ccnnc4)=O)C2)C3)cnc(O)c2cncn12 68579,Cc1csc(=NCC(=O)N(C2CCCN(C(C3CS(=O)(=O)CC(=O)N3)=O)C2)C)[nH]1 68580,N1(C(=O)Cc2cscn2)CCN(C(C2CC3(CCC3)CO2)=O)C(c2cn[nH]c2)C1 68581,N1(C(C(=O)Nc2ccc(C(=O)OC)cc2)C2CC2C)C2CCC1CC(F)(F)C2 68582,c1(NCC2CCN(CCC)C2)[nH]c(=NC(C)c2cn[nH]c2)nc2sccc12 68583,Cc1cc(C(=O)NCC2CC(NC(C3(C)CSC3)=O)C2)c(Cl)cc1Cl 68584,C1(NC(=O)NC)CCC12CCCO2.c1(CNC(=O)OC(C)(C)C)c[nH]nc1CO 68585,c1(N2C(C)(C)C(NC(=O)Cn3cncn3)CC2)cc(C#N)ccc1[N+](=O)[O-] 68586,N1(C(c2ccn(CCC)n2)=O)CCN(C(c2cc(CN(C)C)on2)=O)CC1CF 68587,C(C)(CC(C)NC(c1ccnn1C1CC1(F)F)=O)NC(COCCOCC)=O 68588,c1(C(N2CCCC(C(C)NC(C3(SC)CCC3)=O)C2)=O)cc(C)nc(O)c1 68589,N1(C(C2C(CCOC)C2)=O)CCN(C)C(C(=O)NCC2(CO)CC3CC3C2)C1 68590,Cc1ccc(F)c(C(N2CCN(C(=O)Cn3nc(Cl)ccc3=O)CC2)=O)c1 68591,Cc1[nH]c(C#N)cc1C(=O)NC(c1nocc1C(=O)NCCOCC(F)F)C 68592,C1(C(N2C(C(C)NC(Cn3c(C)c(Cl)cn3)=O)CCC2)=O)CCn2nccc2C1 68593,N1(C(c2scc(C)c2C)=O)C2CCCC1CC(NC(C1C=CCCC1)=O)C2 68594,N1(C(C(CC)O)=O)CC2(CCC2)CC1CNC(c1ccnc(-c2ccco2)c1)=O 68595,Cc1cc(C)n(CC(=O)NCCC2(O)CCN(C(c3[nH]ccc3C)=O)C2)n1 68596,C1(C(=O)NC(C2(C(=O)OC)CC2)C)C=CCN(C(=O)CC23CCC(CC2)C3)C1 68597,N1(C(CC(C)=C(C)C)=O)CCCC(C)(C(=O)Nc2cccc(Cl)c2)C1 68598,C(CC)(CCCC(=O)N1CC2COCC2(CO)C1)NC(C(CC)O)=O 68599,C12CN(CC1F)C2=O.c1(CNC(C(=O)OCC)=O)ccc(N2CCNCC2)cc1 68600,Cc1cccc2c(C(=O)NCC34CC(NC(=O)Cc5ccn(C)n5)(C3)C4)coc12 68601,CCC(F)(C(=O)OC)C(=O)NCCC12CCC(CC1)N(C(c1cn[nH]c1)=O)C2 68602,Cc1cncc(C(N2CCC(CNC(c3nncs3)=O)C2)=O)c1 68603,C1(N(C(c2c(CC)[nH]cc2)=O)C)CCN(C(=O)C=Cc2cncc(O)c2)CC1C 68604,c1(C(N2CCC(N(C(COCC(C)C)=O)C)C2)=O)cc(N)cc(F)c1 68605,CCCCC(O)CC(=O)N1CC2C(CNC(=O)C=C(Cl)Cl)C2C1 68606,Cc1ccc(F)c(CNC(C2(CNC(C3CCSC(C)C3)=O)CCOCC2)=O)c1 68607,C1(NC(C(C)SCc2ccccc2)=O)CCN(C(c2cc[nH]c2)=O)CCC1CO 68608,c1(NC(C2(NC(CC3(C(=O)OC)CC3)=O)CCC2)=O)ccc(OC)cc1F 68609,N1(C(C2C(C)(C)C2)=O)CCCC2CCN(C(=O)C=Cc3nccs3)CC12 68610,C1(NC(COCc2c(C)ncs2)=O)CCCN(C(c2cccc(F)c2F)=O)C1C 68611,C1(NC(C2(C)CC2c2ccc(Br)cc2)=O)CCSC2(C1)CC(C(N)=O)C2 68612,C(CCCCN1CCCC1)NC(C(c1ccccc1)NC(=O)NC1CCCO1)=O 68613,Cn1cc(C(=O)NCC2(NC(=O)CC3=CCOCC3)CC2)c2ccccc12 68614,CC(c1ccccc1F)=CC(N1CC(N(C)C(C2COCCN2C)=O)C1)=O 68615,C1(CNC(C2(C(C)C)CCOCC2)=O)CNCC(C)(C)C1 68616,N1(C(CCCN(C(C)=O)C)=O)CC2CCC1CC2NC(C1CCC(C2CC2)O1)=O 68617,C1(C(CO)NC(C2(NC(=O)COCC3CCC3)CC2)=O)CCCCC1 68618,c1(NC)ccc(C(=O)NC2CCC2NC(=O)CCc2ccncc2)cc1[N+](=O)[O-] 68619,C1(C(=O)NCC2(COC)CN(C(C3COCCN3C)=O)C2)CC2CCC(C1)S2 68620,c1(C2CCN(CC(=O)NC(C(=O)OCC)CC)C2)c(C)noc1C 68621,C1(NC(=O)CC2(O)CCC2)CC2CCC1CN2C(C1CNC(=O)N1)=O 68622,C#CCCC(C(=O)Nc1cccc(C#N)c1)NC(c1[nH]nnc1C)=O 68623,C(=O)(CC(C)CC(C)(C)C)NCCC(=O)NCc1ncc(C)cn1 68624,Cc1ccc(C(=O)NC2CCOCC2NC(C23CC(F)(C2)C3)=O)c(F)c1F 68625,N1(C(CCCOC(C)=O)=O)CCC2CCCC12C(=O)N(C1CCC(=O)N(C)C1)C 68626,C1(C(=O)NCC23C(CN(C(CNC(=O)OC)=O)C2)C3)CCc2nc(C)[nH]c2C1 68627,Cc1nc(CC(=O)NCC2C3CN(C(=O)CCc4ccccc4F)CC23)oc1C 68628,c1(C(N(C(C(=O)NC(CCC)c2nn[nH]n2)C)C2CC2)=O)snc(C)c1N 68629,CN1CCC(NC(=O)C(C2(C)CC2)NC(c2cc3n(n2)CCC3)=O)C(C#N)C1 68630,C(=O)(C(C(C)O)NC(C)=O)NCCN(C(c1cc(C2CC2)ns1)=O)CC 68631,c1(NC(=O)NCc2ncc(C)s2)c(F)cc([N+](=O)[O-])cc1Br 68632,c1(C(N2CCCC(CCNC(C(C)=CC)=O)C2)=O)cccc2c1OC(C)C2 68633,CCC(C)(C(=O)N1CC(CO)(NC(=O)CCc2nc(O)n[nH]2)C1)OC 68634,N1(C(CCC=CCC=C)=O)CC(NC(=O)C(=Cc2ccccn2)C)CC1(C)COC 68635,CC(C(C)(C)NC(=O)CCC1CC1(F)F)NC(=O)CSCC(N)=O 68636,c1(C(=O)NC(CC2CN(C(c3cc(C)[nH]n3)=O)C2)C)cc2sccc2s1 68637,O=C(C#CC1CCOC1)N1CCCOC(CN=c2cc[nH]c(-c3nccs3)n2)C1 68638,N1(C(C(CC)N(C)C(c2ncnc(C)c2C)=O)=O)CCCC(C)(C)C1C 68639,N1(CC)CC2CCC1CN2C(C1CC(NC(=O)OC(C)(C)C)CCO1)=O 68640,N1(C(C2(CC=C)CCN(C(=O)C(C)OCCC(C)C)C2)=O)CCC(O)CC(C)C1 68641,N1(CC)CCN(C(C2(CF)CCN(C(=O)C=CC(C)C)C2)=O)C(C)C1 68642,c1(COCC(=O)NC2CCCC(N(C)C(=O)C3CC3)C2)ccc(C#N)cc1 68643,N1(C(COCCC)=O)CC(NC(=O)C(C)(C)Cc2cnn[nH]2)CC1(C)C 68644,CCCCCCOCC(=O)NCC1(NC(c2cnc(O)o2)=O)CCOC1 68645,CN1CCC(C(N2CCC(N3CCCC3)C2)C(=O)NCc2ccco2)CC1 68646,c1(OC)cc(C(CO)NCc2cc(Cl)ncc2NC(=O)OC(C)(C)C)cc(F)c1 68647,C1(NC(C2CCCC2O)=O)CN(C(=O)C2=CCCOC2)C2(CCC2)C1 68648,C1(COCC#C)CCCN1C(=O)C(C1CCC1)NC(=O)C(C)NC=O 68649,C1(C2CC2)(CNC(CN(C2CC2)CC)=O)CCN(c2nc3ccccc3o2)C1 68650,c1(C(=O)NC2CCC(NC(CCNC(N)=O)=O)CC2)cc2ccc(Cl)c(F)c2[nH]1 68651,N1(C(CC(=C)C)=O)CCCC2CN(C(C3CCc4c(nnn4CC)C3)=O)CCC12 68652,C1(C#CC(=O)NC23CC(C(N4CCC(c5cnco5)C4)=O)(C2)C3)(CC)COC1 68653,N1(C(c2nn(CC)c(O)c2)=O)CC(NC(=O)C=CS(C)(=O)=O)CC2(CC2)C1 68654,Cc1cccc(C)c1C(=O)NC(C1CCCN(C(=O)CC(C)(C)C#N)C1)C 68655,c1(CC(=O)NC2CCCC2NC(c2nsnc2O)=O)c[nH]c2nccc(Cl)c12 68656,Cn1c(O)nc2cc(C(=O)NC3CN(c4cnc(C#N)cn4)CC3(C)C)ccc12 68657,Cc1noc2ncc(C(=O)NC3CC4CC3N(C(c3ncccn3)=O)C4)cc12 68658,CC1(C)CC(O)(CC(N2CC(CCCCNC(c3nn[nH]c3Cl)=O)C2)=O)CO1 68659,c1(NC(c2c(C)cccc2)CO)cc(Br)ccc1S(=O)(=O)NCCC1CCCC1 68660,Cc1ccc(CNCc2cncc(-c3cc(Cl)cc(Cl)c3Cl)c2)c2cccnc12 68661,C(=O)(CC(C)CC(F)(F)F)NC1(CNC(C2ON=C(C(C)C)C2)=O)CCCCC1 68662,Cc1cc(C(=O)NC2CN(C(C3CCOC(=O)N3)=O)CC2F)oc1C 68663,C(=O)(C1=CC2C=CC1C2)N(CCC(=O)Nc1cccc2c1OCC2)C1CC1 68664,C1(NC(CN(C(C)=O)C)=O)CCC(C)(CNC(=O)Cc2csnc2C)C1 68665,C1(=CC(=O)NC(CCC)CCCNC(=O)C(C)CF)CC2CCC(C1)N2C 68666,C#CCCCCCCC(=O)NC1CC(NC(c2ocnc2CC)=O)CC1O 68667,N1(CC#CC)CCN(CC(=O)N(C(C)C)Cc2ccccc2)CC1 68668,C(=O)(C1=CS(=O)CCC1)NC12CCC(CNC(c3cnc(C)[nH]3)=O)(OC1)C2 68669,c1(C(N2C(CCNC(CC3ON=C(C)C3)=O)COCC2)=O)ccc(Cl)cc1O 68670,c1(C(N(C)CC2(NC(=O)CCC3CC3(C)C)CC2)=O)ccnc(Cl)c1Cl 68671,c1(C2(OC)COC2)cccc(C(=O)N(CCC(C)C)Cc2cccc(Cl)c2)c1 68672,N1(c2nccc(=NCC3N(CC)CCCC3)[nH]2)CC(O)C(O)C(O)C1CO 68673,C1(C(N2CCC(O)(CN(C)C)C2)=O)COCCN(Cc2ncnn2C(C)(C)C)C1 68674,c1(NC(N(C2CN(S(N)(=O)=O)C2)CC)=O)ccc(F)c(N2CCOCC2)c1.C(=O)N 68675,c1(C(C)NC(C(=O)NC(C)Cc2cccc(F)c2)=O)ccc(F)c(F)c1 68676,c1(CC(N2CC(F)(CNC(C3(COC)CCCC3)=O)C2)=O)cc(F)ccc1C 68677,C1(NC(C(CSC)(C)NC(c2ccn(C)c2)=O)=O)C(=O)NCCC1C 68678,C1(C2CC2)(C(N2CC(C)(O)C2)=O)CN(C(=O)CCCC2CCCO2)C1 68679,c1(CC(=O)NC2CN(Cc3n(C)nnc3)CC2O)ccc2c(c1)OCO2 68680,CC(C)(C)CC(O)CC(=O)NC1CCCCC1NC(c1cc2cccnn2c1)=O 68681,C(C)(N=c1ccnc(NCC2CC2(C)C)[nH]1)c1ccc(SC)cc1 68682,CCC(C)CCC(=O)NCC(C)(CNC(c1ccc(F)cn1)=O)OC 68683,CCC(CC(=O)N(CC(C)C(=O)NC(c1ccncn1)C)C)C(F)F 68684,C(=O)(C#CC(C)(C)CNC(=O)C(C)CC)NC(CCC)CC 68685,C(=O)(C1=C(Cl)CCC1)N1C(C(C)NC(=O)CCOCC(F)F)CCC1 68686,C1(n2cc(C(C3CC(=O)NC3=O)C)nn2)CCN(C(=O)CC2CCCOC2)CC1 68687,CCCCC(C(=O)NCC1(CC(C)C)CCC1)NC(c1cn(C)nn1)=O 68688,CC(C)CCCC(C)C(=O)N1CCC(C)(C(=O)NCC23CCCC2OCC3)C1 68689,N1(C(CN(C2CCC2)C)=O)CCN(C(C2CC23CCOC3)=O)CC(O)C1 68690,Cc1c(C(N2CC3CC3(NC(=O)CC3CC4(CCC4)CO3)C2)=O)cncc1N 68691,C=CCCCCCC(=O)NC1(C2CC2)CCN(C(c2ccc[n+]([O-])c2)=O)C1 68692,N1(C(c2c(C)ccc(=N)[nH]2)=O)CC2CCCC2(NC(=O)CCC2CCOC2)C1 68693,C1(CC(=O)N(CC(C)NC(=O)CCCCc2cnc[nH]2)C)C(C)(C)C1(C)C 68694,N1(CC(=O)NC2CN(C(C3(C(F)F)CCCO3)=O)CC23CC3)CCS(=O)(=O)CC1 68695,C1(CN(C(=O)COc2cn[nH]c2)CCO)COCCN1CC(F)(F)F 68696,Cc1cc(=N)[nH]cc1C(=O)NCC1CC1CNC(=O)C(C)(C)C(C)C 68697,c1(CC)nc(C(=O)NCCC2CCN(C(C3(CC)COC3)=O)C2)c(C)o1 68698,N1(C(c2c(CC)nco2)=O)CCC(NC(c2ncccc2OC(C)C)=O)C(C)C1 68699,C(C1=NOC2CN(C(=O)CCCc3ccccc3)CC12)NC(CCC=C(C)C)=O 68700,N1(C(CC2C(=O)OCC2)=O)CC(O)(C2CCN(C(=O)CCC3CC3)CC2)C1 68701,C(C(C)(O)C(=O)N1CCCC(CCCCNC(C2CC(Cl)(Cl)C2)=O)C1)OC 68702,C1(C(C)NC(C2CCCC2)=O)CN(C(=O)CCCNC(C2CCC2)=O)CC12CC2 68703,N1(C(c2c(NC)nsn2)=O)CC2=C(C1)CN(C(=O)CC1C=NN(C)C1=O)C2 68704,c1(NC(=O)Nc2cc(C)sn2)cccc(CC2CC2)c1 68705,C1(NC(C(C)(C)NC(C=COC)=O)=O)CN(C(c2cnc(C(C)C)s2)=O)CC1F 68706,C1(C)(CC)CCC(C(=O)NC2CC(NC(=O)C3=C(Cl)CC3)C(O)C2)O1 68707,c1(OC)cc(NC(C2(F)CCN(C(c3c(Cl)ccnc3Br)=O)C2)=O)nc(Br)c1 68708,C12(C(=O)NC34C(CN(C(c5ccc(NC)cn5)=O)C3)C4)CC(C)(CCO1)C2 68709,c1(C(N2CC(CNC(COC(C)(C)C)=O)OCC2)=O)ccnc2[nH]ncc12 68710,C(=O)(C#CC1CCCC1)N(CCOCCNC(C(CCC)(F)F)=O)C 68711,C(C(C)(C)CC(=O)NCCOc1ccccc1)NC(C(C1CCC1)OC)=O 68712,C#CC(C)(C)C(=O)N1CCC(CCCNC(C2CCCOC2C)=O)CC1 68713,C1(NC(c2ccc(CCCC)cc2)=O)CN(C(=O)CN(C)CC)C2CCCCC12 68714,N1(C(c2cnc(CC)s2)=O)CC2CC(NC(=O)CNS(=O)(=O)NC)C2C1 68715,c1(C(N2CCC(C(C)CNC(C3CCSC3)=O)CC2)=O)ccc(P(C)(C)=O)cn1 68716,Cc1nn(C)c(C)c1NC(C1CCN(C(c2ccc(C(F)(F)F)cc2Br)=O)C1)=O 68717,C1(NC(C(C2CC2)NC(CCOC(C)=O)=O)=O)CN2CCC1(C)CC2 68718,N1(C(COCCCCC)=O)CCc2sccc2C1CNC(C12CC(CCO1)C2)=O 68719,CC1CN(C(=O)C#CC(C)(C)C)CCC1NC(c1cccc(NS(N)(=O)=O)n1)=O 68720,c1(C(=O)NC(CN(C(=O)Cc2cc(Cl)n(C)n2)CC)C)cc2n(n1)CCCC2 68721,N1(C(CCC2(NC(CSCCC(C)C)=O)CCC2)=O)CCOC(C(C)C)CC1 68722,c1(C(N2CC(OC)C(NC(c3cnc(Cl)s3)=O)C2)=O)cc(C)n(C(C)C)c1C 68723,C(=O)(C1=NOC(C(C)(C)C)C1)NC(C)CNC(=O)CC(C)(C)c1ccc(F)cc1 68724,C1(CNc2ccc(N3C(=O)OCC3)cc2)CC2OC1C1CC21 68725,Cc1cccc(C(N2CCN(Cc3ccc(F)c(F)c3)C(C)C2)=O)c1C 68726,c1(OC)cc(CN(C2CCN(C(C3CN(C)C3)=O)C2)C)c([N+](=O)[O-])cc1O 68727,C(C(C(=O)N(C1CCC1C)C)C(C)C)NC(CCC(=O)NCC)=O 68728,C1(NC(c2cccc(C3CC3)c2)=O)CC1C1CCCN(C(c2cccnn2)=O)C1 68729,c1(OC(C(=O)N(CCN(C(c2cc(CCC)on2)=O)C)C)C)ccc(Cl)cc1C 68730,C1(OC)CC(CNC(=O)CN2CCCCC2)N(C(=O)CN2CCCOC2=O)C1 68731,N1(C(C=CCN(C)CC)=O)CC2CCCC2(CNC(=O)CCCCN(C)C)C1 68732,c1(C(N(C2CCCN(C(C3CCCC4CC34)=O)CC2)C)=O)nc2ncccn2n1 68733,N1(C(CC(=C)C)=O)CCC(CCNC(c2cncc(NS(C)(=O)=O)c2)=O)CC1C 68734,c1(OC)ccc2oc(C(N3CC4CC3C4C(=O)Nc3ccc(O)nc3)=O)cc2c1 68735,c1(OCC(=O)NC(C(C)(C)C)C(=O)NCC2CSC2)ccccc1[N+](=O)[O-] 68736,N1(C(CCCC#C)=O)CCn2cc(C(=O)N(CCCC)CCOC)nc2C1 68737,CC1CC(CNC(=O)C(C)(C)N2CCCCC2)CN1C(=O)C(C)N(C)C 68738,O=Cc1cccc(CN2CCC3(CC3C(=O)Nc3ccc4c(c3)OCO4)C2)c1Br 68739,C1(C(=O)NC(C(=O)NCCC2CC=CC2)c2cccs2)(C2CC2)CCCO1 68740,c1(CS(=O)(=O)N(c2nncs2)CCC)cccc(F)c1 68741,N1(C(c2c(C)c[nH]n2)=O)CC(C)(C)C1C1CCN(C(=O)C(=O)NC2CC2)CC1 68742,C12(NC(c3n(C)ccn3)=O)CCC(CC1NC(C1CC1c1ccc(F)cc1)=O)C2 68743,C1(NC(CC2N(CC)CCOC2)=O)CCN(C(c2cn(C)nn2)=O)CC(C)(C)C1 68744,C1(CC(=O)OC)(NCC(c2ccc(C)cc2)O)CS(=O)(=O)C1 68745,c1(CN2CCC(NC(c3cnc(O)nc3O)=O)CC2)c(Cl)cc(Cl)cc1Cl 68746,C(=O)(C1=NOC2COCC12)N1C2C(NC(CCNC(N)=O)=O)CC(C2)C1 68747,c1(CNC(COCC(C)C)=O)nc(CNC(=O)C(C)(C)c2cncs2)cs1 68748,CC1CCN(C(C2CCCC2(C)C)=O)CCN1C(c1cnco1)=O 68749,CCCCC(CC)C(=O)NCC(CCCC)NC(C1CC(F)C1)=O 68750,n1(CC(=O)N(C(c2ccccc2)CNC(c2cnnn2C)=O)C)nnc(C2CC2)n1 68751,C(CCCCCNC(c1c(Br)nnn1C)=O)NC(CC1ON=C(C)C1)=O 68752,C(CCCC(=O)OC)(C(=O)NCc1cccc(Br)c1)N1CCCC(COC)C1 68753,C(=O)(C(C)CC(C)C)NCc1c(C(=O)NC(CCCC)(C)C)occ1 68754,Cc1cc(CNC(=O)C(=O)N(C)CCOCCOCCO)c(C)o1 68755,C(=O)(C1CCc2c(Cl)cccc21)N(C(Cc1ccc(C)cc1)C(=O)O)CCOC 68756,N1(C(c2cc3ncccc3o2)=O)CCC2(CCCN2C(c2c[nH]c(=O)cn2)=O)C1 68757,CC1=CCCN(C(=O)NCCCC2CCCO2)C1 68758,S(=O)(=O)(c1cn(-c2ccccc2)nn1)NCC1(CO)C(C)(C)C1 68759,C(=O)(C(O)CC(F)F)NC(C1CCN(C(=O)C(C)(C)c2cnco2)CC1)(C)C 68760,C1(C(=O)NCCC(=O)NC(CC)C)CCOCC1NC(C1OC2CCC1C2)=O 68761,c1(C(=O)NC2C(CNC(C3(Br)C(C)(C)C3)=O)C2)ccn2c(O)nnc2c1 68762,C(C(COC)C(=O)NC(CO)C(C)NC(C1(N(C)C)CCC1)=O)OC 68763,c1(N2CCC(OC(c3c(C)nc(CC)s3)=O)C2=O)ccc(Cl)cc1F 68764,C12(COC)CC(CNC(c3ccc(Cl)o3)=O)(CN1C(C1(C(F)F)CCCO1)=O)C2 68765,C1(NC(C2(CCNC(C(CC)(C)C)=O)CC2)=O)CC2CC1C(O)C2O 68766,C1(CNC(CC2(OC)CCC2)=O)CN(C(C2(C)CSC2)=O)CCC1C 68767,N1(C(c2ccc(C3CC3)nc2O)=O)CC2CCCN(C(=O)Cc3cccs3)C2C1 68768,Cc1cc(C(=O)NCC(C)CN(C)C(c2c(C(F)F)cnn2C)=O)sc1C 68769,C(C(=O)NCc1cn(C2CN(C(=O)CC(C)C)C2)nn1)(C(C)(C)C)NC(C)=O 68770,N1(C(C(C(C)CNC(c2coc3c2COC3)=O)F)=O)CCCCN(C)CC1 68771,c1(-c2scc(CC(=O)NCCN(C(c3c(CC)nco3)=O)C)n2)ccc(O)cc1 68772,Cc1cc(C(=O)NCC(C)(C(C)C)NC(=O)CC2CCCC(C)(C)O2)nc(O)c1 68773,C1(NC(C2C(OCC)C2)=O)CN(c2nnco2)C1 68774,c1(C(=O)NC2C(NC(c3sc(CC)c(C)c3)=O)CC2)ccc(F)c(F)c1C 68775,C1(C(=O)NCCN(C(CN2CCN(CC)CC2)=O)C)CC(C2CCCC2)C1 68776,c1(C(N(CCOC)CCNC(=O)Cn2cnccc2=O)=O)cc(O)cc(N)c1C 68777,C(=O)(C(CCNC(c1ccc[n+]([O-])c1)=O)OC)N(C)CC1(OC)CCCC1 68778,C=CCC(C)C(=O)NC(C1(C(=O)NC(CCOC)C(C)C)CC1)C 68779,N1(C(CSSC)=O)CCC2(CCCCC2NC(c2nncs2)=O)CC1 68780,N1(C(CCCCCNC(CCCCC=CC)=O)=O)CC2CC(C)(C)C2C1 68781,O1C=CC(O)(C(F)(F)F)Cn2cc(nn2)C1.C(=O)(C(C)(C(C)C)NC)N(C)CC 68782,c1(OC)c(C(=O)NCC2CC2NC(C2CC2CC(C)C)=O)cccc1Br 68783,Cc1cc(C(N2CC(NC(C3C4COCC34)=O)C(n3cccn3)C2)=O)nc(C)n1 68784,C(C)(CNC(C1(C)CC1(F)F)=O)(CC(C)C)NC(C=CCCC)=O 68785,Cc1nc(C(C)C)nc(O)c1C(=O)NC1CCCC1NC(C1(CF)CC1)=O 68786,CC(=O)CCCC(=O)N1CCC(C(F)(F)F)C(NC(=O)Cn2nc(C)cc2N)C1 68787,C#CC1CCCC(NC(C2CC(F)(F)CN2C(=O)CCOCC(F)F)=O)C1 68788,N1(C(Cc2cnc(C)[nH]2)=O)CC2CCC2(CNC(C2CC2C(C)C)=O)C1 68789,N1(C(C(C)NC(N)=O)=O)CC(CNC(=O)Cn2nccn2)C(c2ccccc2)C1 68790,C(=O)(C1=NOC2COCC12)N1CC=C(C(=O)NCCC(C=C)C)CC1 68791,c1(CC(N2CC(OCCNC(COCCC(C)C)=O)C2)=O)ccc2ccoc2c1 68792,C1(CCNC(C(CC)(F)F)=O)C(C)CCCN1C(=O)CCOc1cccc(F)c1 68793,C(CSC1CCCO1)(C(=O)NC1CC1NC(=O)CSC(F)(F)F)OC 68794,S(=O)(=O)(c1cccc(Br)n1)N1C(C)(C(=O)NCc2cncc(Br)c2)CCC1 68795,C1(NC(C(CCC)C)=O)CCC12CCN(C(c1c[nH]c(=NC)s1)=O)CC2 68796,C1(NC(C2(SC)CC2)=O)CCCC2CN(C(c3noc4cc(F)ccc34)=O)CC12 68797,N1(C(c2c[nH]c(=N)o2)=O)CC(CNC(c2cccc(-n3cccn3)n2)=O)C2CC12 68798,CCCCCCC(=O)N1CCCC1CNC(c1cccc(Cl)c1OC(F)(F)F)=O 68799,C1(OC)COc2c(C(N3CCCC3CN(C)C(c3scnc3Cl)=O)=O)cnn2C1 68800,O=c1cc(C(F)(F)F)oc2c(NCCC3CCCCO3)cccc12 68801,Fc1ccc(Br)c(Cn2cc(C3CCC3)nn2)c1 68802,c1(OC)ccc(C(=O)NCC2CC(C)N(C(=O)CCc3cnccn3)C2)cc1Cl 68803,c1(C(=O)NC2CC(C(N3CCC(C4CCCO4)C3)=O)C2)ccnc(CO)c1 68804,Cc1nc(Cl)nc(N2CCC(NC(C3CCCC(F)(F)CC3)=O)CC2)c1[N+](=O)[O-] 68805,CC(C)(C#N)CCC(=O)NC1(CNC(c2cc3ccccc3o2)=O)CCOC1 68806,C1(C(C)C)CN(C(C2(Cl)CC23CCC3)=O)CCN1C(c1sccc1CC#N)=O 68807,C1(C(NOCC(CC)C)=O)CCC(C)N1C(c1ccc(C)n1C)=O 68808,c1(C(=O)NCC2C(NC(C3CC=C(C)CC3)=O)C2)cn(C)cc(Br)c1=O 68809,C=CC(C)(C)CC(=O)NC1(CNC(=O)COCc2ccnn2C)CCCCC1C 68810,c1(C(=O)NC2CCN(C(C(C)n3cnnn3)=O)CC2)cc(Cl)c([N+](=O)[O-])cc1F 68811,CC1=NOC(C)(C(N2CC3C(NC(c4cn(C(F)(F)CO)nn4)=O)C3C2)=O)C1 68812,c1(C(c2ccccn2)NC(c2ccc(C3CC3)cn2)=O)ccccc1F 68813,CC1CC(NC(C2(F)CC2)=O)CCN1C(c1ccc(-c2ccccc2)cc1F)=O 68814,c1(NCC(=O)NCCC(C)NC(C2C3CCCC23)=O)ccc(Cl)cc1Cl 68815,C(C(O)C(=O)NCCN(C(=O)C(C)N(C)C)CCSC)SC 68816,C1(CC)CN(C(C2CC3CC3CC2C)=O)CCN1C(c1ccccc1CC#N)=O 68817,C1(CCNC(C(C)=CC2CC2)=O)CCN(C(c2cc(C3CCCC3)no2)=O)CC1 68818,CCC(CCCC(=O)NC1(C)CCCC1(F)F)NC(c1c(C)ccn1C)=O 68819,C#Cc1ccc(CC(N2CCC(F)(C(N3CCC(F)(CO)C3)=O)CC2)=O)cc1 68820,C1(C(=O)NC(C)CC2CCOCC2)CC(F)CN1C(=O)CCOC1CCCC1 68821,C=Cc1ccc(C(=O)NC(C)C(C)C(=O)N(CC(C)C#N)C2CC2)cc1 68822,n1(CCOC)ccc(=NC(=O)C(=O)NCC2Cc3ccccc3C2C)[nH]1 68823,c1(C(=O)NCCNC(c2cn(CCN(C)C)nc2)=O)cc(S(C)(=O)=O)ccc1F 68824,c1(C(=O)NCC(=O)NCCC(C)NC(c2cccc(=O)o2)=O)ccc(N)cc1 68825,C(C)(C)(C(C)CC(=O)N1CCC2CC12)NC(CC(C)CN(C)C)=O 68826,Cn1c(NCC2CC(NC(=O)CN3CCCC3=O)C2)c(C#N)c(=O)n(C)c1=O 68827,CCCC(C)CC(=O)NCCN(C(C1(c2ccccc2C)CC1)=O)CC 68828,C1(CCC(=O)NC2(COC)CCC2)CCN(C(=O)CCn2ccnn2)C1 68829,Cc1cc(C(N2CCCC(NC(=O)CN(C)C3CC3)C2)=O)c(F)cc1N 68830,C1(NC(c2scc(OC)c2OC)=O)CC2(C1)CN(C(C1CCOC1(C)C)=O)C2 68831,C1(OC)CCC2(CCN(C(c3ccc(CNC(=O)C4=CCOCC4)s3)=O)C2)C1 68832,c1(C(N2C(C(N3CC(C=C)C(O)C3)=O)C(C3CC3)CC2)=O)cccc2ccoc12 68833,c1(COC)csc(C(N2CCC(CNC(C3CC3(Cl)Cl)=O)C2)=O)c1 68834,C(=O)(CS(=O)c1ccc(Cl)cc1)N1C(C(C)C)CN(C(=O)COCCSC)CC1 68835,c1(C(C)(C)C)ccc(C(N2CCCC(N(CCO)C(c3cscc3Cl)=O)C2)=O)cc1 68836,CN1CCN(C(C2CC(C)(C)C2)=O)CC1CNC(=O)C(c1ccc(C#N)cc1)O 68837,C1(CNC(C2CC23CCC3)=O)CC(C)CO1.CC(C)(C)OC(=O)NCC(=O)O 68838,Cc1cc(Cl)n[nH]c1=NC(=O)C1CC(O)CN1C(c1cccc2c[nH]nc12)=O 68839,N1(C(CCCN(C)C)=O)CC2(CC(NC(C3(N4CCOCC4=O)CC3)=O)CO2)C1 68840,C1(C)(NC(C2CC(=O)N(C)C2c2ccccc2)=O)CCc2ccccc2C1 68841,n1(CCC(=O)NCCOCC(=O)NCC(C)(C2CC2)OC)ccnc1C 68842,N1(C(C(CC)C)=O)CCC(NC(=O)CN(C2CCCC2O)C)C1C 68843,Cc1ccc(C)c(CC(=O)NCC(C2CCN(C(c3occc3C)=O)CC2)C)c1 68844,C1(C(C)(C)NC(C2CCC(C)S2)=O)CCN(C(=O)CCc2cccnc2)CC1 68845,N1(C(CCN(C)CC)=O)CCC(C)(CCNC(C2CCC(F)C2)=O)CC1 68846,C1(CNC(CCOCC)=O)CN(C(=O)C(c2ccccc2)NC(N)=O)CC1O 68847,CON1CC(C(=O)NC2CCCCC2NC(=O)CC2CC2)CC1=O 68848,C1(NC(=O)Cn2ncnn2)COC2(C1)CN(C(c1cc(C(F)(F)F)on1)=O)C2 68849,CC1(NC(C2CC2C(F)(F)F)=O)CCCN(C(C23CC4CC2C3C4O)=O)C1 68850,C(C)(C)(CCCCC(=O)NC1CCC(NC(c2cscc2OC)=O)C1)OC 68851,C(CC1CC1)(C(=O)N(CCCO)CC)NC(CNC(=O)OCC=C)=O 68852,c1(C(=O)NCCCOCCNC(CSCC#C)=O)nnn2c1CCCCC2 68853,C1(F)(C(N2CCN(CC(C)NC(c3cc(C)no3)=O)CC2)=O)CCC(C)CC1 68854,c1(C(=O)NCC(CNC(=O)C(O)C(F)F)OC)cc(F)c(F)c(F)c1 68855,N1(C(c2ccc(C#C)cc2)=O)CCC(C(=O)NCCN(CC(F)F)C)CC1(C)C 68856,c1(SCC(=O)NC(CNC(c2nc(C(C)OC)oc2)=O)C)ccccc1O 68857,C(=O)(C#CC1CC1)NCc1c(C(=O)NCc2c(COC)ocn2)scc1 68858,C(=O)(C(C(=O)NC(C1CCCCC1)CNC(=O)Cc1cncn1C)OC)OC 68859,C(Cc1cn(-c2ccc(N)cc2)nn1)(CC(=O)O)NC(c1ccn(C(C)C)n1)=O 68860,c1(C(=O)NC2CC(NC(CCSC)=O)C2(C)C)ccc(NS(C)(=O)=O)cc1O 68861,c1(C(=O)NCc2cc(OC(CC)C)ncc2)c(C)cc(Br)cc1F 68862,C1(CNC(C(CC)C)=O)CCCCN(C(=O)CCc2ccc(O)cc2)C1 68863,c1(C(=O)NCCN(C(COc2cn(C)nc2)=O)CC2CC2)cccc(C#N)c1Br 68864,c1(-c2ccc(-c3nccc(O)c3)cc2)c(F)ccc(O)c1F.CO 68865,c1(CNC(C(Cc2ccccc2)OC)=O)cccc(NC(C2CC=CCO2)=O)c1 68866,C1(C(=O)NCCCCCCN(C(C(CC2CCC2)OC)=O)C)CC2CCC1CC2 68867,C12(C(=O)OC)CCCC(NC(=O)NCC3CC(O)C34CCC4)(C1)C2 68868,C(CC(C)C)(C(=O)NCc1ncc(C(=O)NC(CO)CC(F)(F)F)cn1)OC 68869,CN1CCC(C(=O)N(C)CC2CC(F)(F)C2)(NC(=O)Cc2cnn(C)c2)C1 68870,Cc1[nH]nc(Cl)c1C(c1nnnn1C)NC(c1cncs1)C 68871,C1(NC(C2C(CC)CCC2)=O)CC12CCN(C(=O)CCc1ccccn1)C2 68872,N1(C(CC2CC(SC)C2)=O)CC2CCC1CC2NC(c1ncnc(C)c1C)=O 68873,C1(C(N2CCC2(C)C(=O)NC)=O)(CC)CCCN(C(c2ccsc2C)=O)C1 68874,c1(C(=O)NCC2C(NC(C3(C(=O)OC)CCCC3)=O)COC2)ccc(OC)nc1 68875,N1(C(c2c(OC)scc2)=O)CC(C(=O)NCC2(C)CCC2)C(C(C)C)C1 68876,Cc1cnc(CCC(=O)NCC2CCCN2C(c2nncn2C(C)C)=O)[nH]1 68877,c1(C(=O)NC2CCC(NC(C3N(C(CC)=O)CSC3)=O)C2)cnccc1Cl 68878,Cc1cc(NCC(c2cc(F)ccc2F)=O)cc2c1CCC2.C1C(=O)N1 68879,c1(C(=O)NCc2ccc(C(N(C)Cc3nc(=O)o[nH]3)=O)s2)cc(C#N)cn1C 68880,c1(CCOC(C)C)ccc([N+](=O)[O-])cc1.c12ccccc1-c1cc(ccn1)NC2 68881,C(CC(=O)NCC1CCN1C(C1CC(=C2CC2)C1)=O)(C(F)(F)F)OC 68882,O=C(C1=C(Cl)CCC1)NC(Cn1ccnn1)C(N1CC2(CCC2)C1)=O 68883,CC1CCCN(C(c2c[nH]nc2C(F)F)=O)C1CCNC(c1ccc(C#N)[nH]1)=O 68884,C1(C2CCCCO2)(C(N(C)CC2CC2)=O)CCCO1 68885,C1(CC)CCCC1C(=O)NCc1ccc(C(=O)NCCCC2(O)CC2)o1 68886,C1(C(=O)NCC(=O)NC(C)C)CCN(C(=O)COc2ccn(C)n2)C1C(C)C 68887,c1(N(CC2CN(C(=O)OC(C)(C)C)C2(C)C)CCO)ccnc(Br)c1N 68888,C1(=O)CCCC(C)N1.C1(C(=O)NCCCN(CC)CC)(OC)CCOC1 68889,c1(C(N2CCC(CNC(Cc3scc(C)c3)=O)C2)=O)ccnc(C)n1 68890,N1(C(C(=Cc2ccccc2)CC)=O)CCOCC(CNC(=O)C=NOC)C1 68891,c1(CC(=O)OCC2CC2c2ccccc2)ccc(N2CCCC2)cc1 68892,C1(CC(N2CCN(C(C(C)OC)=O)C(C)C2)=O)SC2=NCCN2C1=O 68893,c1(C(=O)NCC#CCNC(CCCc2onc(CC)n2)=O)ncnc(O)c1Br 68894,c1(SCC(N2CCC(CNC(C(CC)F)=O)CC2)=O)ccc(F)cc1F 68895,C(=O)(CC(C)CC(=O)OC)N(C(CC)C(=O)NC1COCC1O)C1CC1 68896,c1(NC(CC2N(C(c3cc(C)[nH]c3)=O)CCC2)=O)ccccc1C(C)(C)O 68897,c1(N2C(C)CC(CNC(c3csc4ccccc34)=O)C2)ncnc2c1ncn2C 68898,C=CCC(CC(C)C)C(=O)N1CC2(C1)CN(C(C1CC(O)CN1C)=O)C2 68899,C12(C(N3C(CN(C)C(c4cnc(Br)s4)=O)CCC3)=O)CCC(C)(C1)OC2 68900,N1(C(C(CCSC)OC)=O)CCCC(C)C1CNC(=O)COC1CCCCC1 68901,c1(C(=O)NCCCCC2CN(C(C3CCC(C)O3)=O)C2)c(F)cccc1F 68902,N1(C(C2CCc3nnc(O)n3C2)=O)CCC2C(CCCN2C(C2CC(F)C2)=O)C1 68903,C(=O)(C(=O)N=c1ncn(Cc2ccccc2)[nH]1)NC1C(C)C2CCC1C2 68904,Cc1ccc(CNC(=O)CC2(CNC(C3CCC3C)=O)CC2)cc1F 68905,C1(SC)CCCN(C(=O)CSc2nccn2C)CC1.C1(=O)C(C)N1CC(F)(F)F 68906,C12(NC(C(C)OC)=O)CCCC1N(C(=O)CC=CC(C)(C)C)CC2 68907,CN1CC(C)(C)CC1C(N1CC(CCO)(NC(=O)Cc2cc(F)cc(Cl)c2)C1)=O 68908,C=C(C)C1OCCC1CNC(=O)CN(C(=O)Cn1ccc(C)n1)C1CCC1 68909,Cc1ccc2c(C(=O)NCC(C)(C)NC(C34CCCC3CS4=O)=O)onc2c1 68910,c1(OC)cc(C(F)(F)F)ccc1-c1cc(CN2CCC(Br)CC2)ccn1 68911,C(=O)(C(F)(F)F)NCC(=O)NCCN(C(=O)Cc1cccn1C)CC 68912,C=CC1CN(C(=O)C(C)S(N)(=O)=O)CC1NC(C1(CC2CC2)CC1)=O 68913,c1(C(N2C(CNC(c3ccoc3Cl)=O)CCC(C)C2)=O)cccc2c1ncn2C 68914,C1(NC(CCc2onc(C)n2)=O)COCCN(C(C2COC(=O)N2)=O)C1 68915,N1(C(C2C(COC)CC2)=O)CCCC(O)(CNC(c2cn(C)nc2C(C)C)=O)C1 68916,O=C(NNc1cccc2c1OC(F)(F)O2)c1c(Br)ccc(F)c1I 68917,c1(C(N(CCCN(C(c2c(C)sc(O)n2)=O)C)C)=O)cnc(Cl)c(N)c1 68918,N1(C(C(C2CCCC2)OC)=O)CCCC2(C1)CN(C(=O)COC1CCCO1)C2 68919,C12(C(=O)NCC3(CCNC(C(C4CC4)OCC)=O)CC3)CC(C)(C1)OC2C 68920,C12(C(=O)NCC(CNC(C3(CS(N)(=O)=O)COC3)=O)O)CCCC(=O)N1CCC2 68921,C1(NC(C2(CC(C)C)CC2)=O)CC2CCC(C1)N2C(C1CCCCC1(C)C)=O 68922,N1(C(C=C(CCC)CCC)=O)CC(C)N(C(=O)CC(C)C(F)F)C(C)C1 68923,C1(NC(CSCCOC)=O)CC2COCC2N1C(=O)CCCCN(C)C(C)C 68924,C1(NC(C(CC)NC(N)=O)=O)CC(OC)CN(C(=O)Cc2c(O)ncnc2O)C1 68925,C1(C(C(=O)NCC(CC)O)F)CCN(C(=O)CSC2CC2)C1 68926,Cc1cnc(NC(C2CCN(Cc3ccc(Cl)cn3)CC2O)=O)nc1Cl 68927,c1(NCCN=[N+]=[N-])ccc(C(=O)NC2(CC(N)=O)CCCC2)cc1 68928,c1(CN2C(C)(C(=O)Nc3c(C(=O)OC)c(C)no3)CCC2)c(O)cc(O)cc1O 68929,CC(C)CC(CC(C)C)C(=O)N1CC2(CCCC2NC(c2ccncc2N)=O)C1 68930,c1(SC)cc(C(=O)N(C)CC2CCCN(C(=O)CC3COCC3O)C2)nn1C 68931,c1(CC)nncn1CCNC(=O)CC1CCN(C(=O)CCOCCCOC)C1 68932,N1(C2CN(C(C3C(=C)CC3)=O)C2)CC(NC(C2CN(C(N)=O)C2)=O)CC1=O 68933,Cc1ccc(C(=O)NCCCOC2CCN(C(=O)C3=CCCO3)CC2)nc1F 68934,N1(C(C(C)(O)c2ccccc2)=O)CCC(CO)(NC(c2ccoc2)=O)C1 68935,C(=O)(CCCC(F)(F)F)N1CC(O)(CNC(C23CCCCC2C3(F)F)=O)C1 68936,N1(C(c2cn(CC=C)nn2)=O)CC2CCC1CN2C(=O)C(C)NC(C1CCC1)=O 68937,N1(C(c2snc(OC)c2I)=O)C(CO)CCCC1CO 68938,c1(C(=O)NCC(C(C)C)C(=O)N2CCOCC2CO)ncn2ccccc12 68939,c1(-c2ccc(F)c(C)c2F)cccc2c(C(=O)NC3CC3)c[nH]c12 68940,c1(OC)ncc(C(=O)NC2CCC(NC(c3scc(C)c3Cl)=O)C2)cc1Br 68941,N1(C(CC(=O)N(C)C)=O)CC=C(CC(=O)N2CCOCC(C)(C)C2)CC1 68942,N1(C(c2c(C)noc2C)=O)CC2CC(O)C1C2NC(c1ccc(CO)cn1)=O 68943,C=CC(F)(F)C(=O)NC(CNC(=O)C(CC)=CCCC)C1CCC1 68944,C1(O)(CC(=O)NCC2(C(=O)NCCN(C(C)C)C)CC2)CCCC1 68945,C1(NC(=O)COC2CCCOC2)CC2CC(NC(c3cnoc3C3CC3)=O)CC12 68946,C=CCCC(F)(F)C(=O)NCCOCCN(C)C(c1cn2cc(C)nc2s1)=O 68947,CC1c2nncn2CCN1C(=O)C(c1ccccc1)(C)NC(=O)C(F)C1CCC1 68948,C1(NC(c2n(CC)nc(C)c2)=O)CCN(C(C23CC(C)(CO2)C3)=O)C12CCC2 68949,C=CCCCCCCC(=O)NC1(CNC(c2cc(C3CC3)ccn2)=O)CCOC1 68950,N1(C(c2cc(CN3CCCC3)c[nH]2)=O)CC2(C1)CN(C(C1COC1)=O)C2 68951,C(C(C)(C)CC(=O)NC(C)CCO)NC(Cn1c(C)nc(C)n1)=O 68952,c1(CC)cccc(N(C)C(C2COCC2NC(=O)CCc2ccn(C)c2)=O)c1 68953,N1(CCC)CCCC(C(=O)NC(C)(C)C(C)NC(=O)CC2CC(C(F)F)C2)C1 68954,S(=O)(=O)(c1c[nH]c(=NCCC(C)O)cc1C)NC(CC)C(C)O 68955,CN1CC2CCCN(C(=O)CCn3cc(CCCN4CCOCC4)nn3)C2C1 68956,C1(C(=O)NCC(C(C)C)NC(=O)CCCC2CC2)CCC(C(=O)N(C)C)CC1 68957,CC(C)(C)C#CC(=O)NCC(CC(=O)NCC1OC(=O)CC1(C)C)OC 68958,c1(NC(C23CC(C)C2C3)=O)ccc2c(c1)CN=S2(C)=O.c12csc(n1)CCN2 68959,c1(C(N2CC(C(C)NC(C3CCCN(C(C)=O)C3)=O)C2)=O)c(C)cc(C)nc1O 68960,C1(C(=O)NCCC2(C(=O)NCCCCCO)CC2)(OC)CCC(C)C1 68961,C12(CNC(C(N3CCCCCC3)C)=O)CCC(CC1)N2C(=O)CC1CC1(C)C 68962,c1(CC(=O)NC(CN(C(c2csc(C3CC3)n2)=O)CC)C)ccccc1C 68963,C1(NC(CSC(C)=O)=O)CCCC2CN(C(c3ccnc(F)c3F)=O)CC12 68964,N1(C(C=Cc2nnn(C)n2)=O)CCOCC(NC(C2C3CCCCCC23)=O)C1 68965,c1(CC(C)C)cccc(C(N2CCC(C(C)(C)NC(c3c[nH]c(Br)c3)=O)C2)=O)c1 68966,C(C)(C)(CCCNC(=O)C=CC=C(Cl)Cl)NC(C(CC)n1ccnc1)=O 68967,C1(C)(NC(N(C)CC2(CS(C)(=O)=O)COC2)=O)CCCN(C(=O)OC(C)(C)C)C1 68968,C1(NC(CCC2C(C)(C)C2)=O)C2CC1N(C(c1ccc(O)cn1)=O)C2 68969,Cc1cc(C(=O)N(C)CC2CCCCN2C(=O)C(N2CCSCC2)C)ccc1O 68970,c1(CN2CC3CN(C(=O)COc4ccc(O)cc4)CC32)c(F)c(F)cc(F)c1F 68971,C(CC(C)C)(CC(C)C)NC(CCN(C(=O)CCC1CCCC1)CC)=O.C(C)(=O)O 68972,C(=O)(C(CC(C)C)C(N)=O)NC1N(C(C(CC#C)C2CC2)=O)CCOC1C 68973,N1(C(CSCC(=O)OC)=O)CCCC(CCNC(c2cccn2C)=O)C1 68974,N1(C(Cc2cc(C)nn2C)=O)CCC2CN(C(=O)CCS(N)(=O)=O)C(C)C12 68975,c1(NCc2n(C)nnc2Br)ccc2c(c1)C(C)(C)CC2(C)C 68976,CCCCCCC(C)CC(=O)NC1CCN(C(C2CC(F)(F)C2)=O)C1C 68977,C1(C(N(C(C)C(N)=O)C)=O)CC12CCN(C(=O)Cn1cnnn1)CC2 68978,CC(C)(C)CCC(=O)NC1(c2ccccc2)CCN(C(=O)C2=CCC2)C1 68979,c1(C(=O)NCC2CC(NC(C(C)C3CCCO3)=O)C2)cc(Br)cs1 68980,CC(c1ccc(F)cc1F)=CC(=O)N(CCCCNC(C1CC2CC2C1)=O)C 68981,C#CC1(C(N2CCC(C(C)O)CC2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)C1 68982,C(CN=c1cc(Cl)nc(SC)[nH]1)C1CCCN(C(C2N(C)CCCC2)=O)C1 68983,c1(C(CC)=O)cccc(OCC)c1.N12CCCC(C1)NC2=O 68984,c1(CNC(CCSCC)=O)cccnc1C(N1CCC(CC(C)(C)C)C1)=O 68985,CCC(C)C(CC(=O)NC1CCCSCC1)NC(=O)CC1CC(=O)NC1=O 68986,N1(C(C(C(C)(C)C)OC)=O)CCC2(CC1)CC2CO.c12cn(nn1)CCCC2 68987,c1(OCCCC)ccccc1NC(=O)NCCC1(O)CCOC1 68988,C1(CNC(=O)C2CC2)CC2(CCN(C(=O)CCOc3ccccc3)C2)CO1 68989,C=CCC(C(=O)NC1(C)CC(NC(C2CC2c2ccc(F)cc2Cl)=O)C1)C(C)C 68990,N1(C(C(C=CCCC)O)=O)CCC(O)(CCNC(c2c[nH]c(C)cc2=O)=O)CC1 68991,C(CC(O)C(F)(F)F)NC(CNC(CNC(c1cc(C)[nH]c1)=O)=O)=O 68992,c1(OCC)cc(C(=O)NCC(CNC(=O)CCC(C)OC)CO)ccc1C 68993,CC(CC(=O)N(C)CCN1CCN(C(=O)CN2CCC(O)CC2)CC1)P(C)(C)=O 68994,C(=O)(CCCCCCNC(C(F)(F)F)C1CCCC1)OC(C)(C)C 68995,C1(NC(c2c(CC)noc2)=O)CCCC12CN(C(=O)CCc1cnco1)C2 68996,C(=O)(C(CNC(c1nc[nH]n1)=O)CC(C)C)N(c1ccsc1)CC 68997,Cc1ccc(C(=O)N(C)CC2CCCCN2C(c2nc(C)ccc2C)=O)c(F)c1 68998,N1(C(C(C(=O)OCC)C2CC2)=O)CC(n2cc(CC3OCCO3)nn2)C2(CCC2)C1 68999,Cc1nc(O)[nH]c1C(=O)NC(C)CNC(=O)Cc1ccsc1C 69000,CC1CN(C(=O)Cc2ccccc2O)CC1CNC(c1ncc(C(F)(F)F)s1)=O 69001,c1(C(C(=O)OC)N(C(C)(C)CC)CC(N2CCCC2)=O)ccc([Si](C)(C)C)s1 69002,C1(C(=O)NC(C)CCCNC(=O)COCC2CC2)C(C(F)(F)F)C1[N+](=O)[O-] 69003,N1(C(C2N(C(c3c(CC)nn[nH]3)=O)CCC2)=O)CCC(C)(C2CC2)C1 69004,C=CC(C)(O)CC(=O)N(C(CNC(=O)C(C)Sc1ccccn1)CC)C 69005,N1(CCCCCNC(C(C)NS(C)(=O)=O)=O)CCN(CC2COCCOC2)CC1 69006,CCN=C(NCc1ccc(C2COC2)cc1)N1CCC2OCCCC2C1 69007,C1(CNC(c2cccc(Oc3ccccc3)c2)=O)CC2CCCC(C1)C2 69008,C(C)(C)(CCC(=O)N1CCC(C)(C(=O)NCC2(C)CCC2)C1)N(C)C 69009,C=CC1COCC1NC(C1CSCN1C(=O)C(C(=O)OC)OC)=O 69010,C1(NC(C=Cc2scc(C)n2)=O)CCCC12CCN(C(=O)CCc1cnco1)C2 69011,N1(C(=O)OC(C)(C)C)CCC2CC12CC(N1CCN(c2ccsc2C#N)CC1)=O 69012,c1(C(C)=O)ccc(C(=O)NCC2CCCN2C(=O)Cc2cc(C)no2)cc1 69013,C1(C(=O)NCC(C)NC(C(C(C)C)NC(C)=O)=O)CCc2ncnc(C)c2C1 69014,C1(CNC(c2n(CC)ccn2)=O)CC(C)N(C(c2scnc2Cl)=O)C1 69015,C1(C(=O)NC2C(C=C)CN(C(=O)CC(=C)Br)C2)CCCCCS1(=O)=O 69016,C1(CCNC(CC(CC)C(C)C)=O)CC(N=c2cc(C)nc(CO)[nH]2)C1 69017,N1(C(c2c(C)cn(C)n2)=O)C2CCC(C2)C1CC(=O)NCCOCC(F)F 69018,c12ccc(Cl)cc1NC2=O.Cn1cc(-c2cn(CO)nn2)c(SC(C)(C)C)n1 69019,c1(C(=O)NCCC(=C)CNC(C2OCCC2CC)=O)cccc2c(C)[nH]nc12 69020,C1(N(C(=O)CC2(O)CCC2)CC)CCCN(C(c2ccc(Br)nc2C)=O)CC1 69021,C(=O)(C1c2c[nH]nc2CCC1C)OC(c1ccc(C)c(F)c1)C 69022,C1(OC)CN(C(C23CC(C(F)(F)F)(C2)C3)=O)CCC1NCc1cc(B(O)O)co1 69023,N1(C(C(=O)N(C)CCC2CC2)=O)CCC(C(F)F)(CN)C1 69024,CCCC(C(O)C(=O)NCc1nc(CC)cs1)NC(=O)C(CC)CCC 69025,N1(CCNC(C2(NC(C3CC=CCC3)=O)CCSC2)=O)CCOC1=O 69026,C12(C(N3CC(C)C(CCNC(=O)Cc4cnc[nH]4)C3)=O)CCC(CF)(C1)OC2 69027,C1(NC(COCCC(C)C)=O)CCN(C(=O)CN2CCCC2C)CC1C(N)=O 69028,N1(C(C=Cc2c(C)n(C)nc2)=O)CCCC(NC(=O)CCc2cnco2)C(F)C1 69029,C1(C)(C(=O)NCCNC(c2cc(SC)oc2)=O)CCCCCC1 69030,c1(C(=O)NCCN(C(=O)CC2(O)CCCC2)CCC)ncc(C(C)(C)C)o1 69031,C1(CC(=O)NCCCOC=C)CCN(Cc2cn(C)nn2)C1 69032,CCCCCCC(=O)NC(CCOCCO)C(=O)N1CCC(CC2CC2)C1 69033,c1(C(=O)NCCCC(C)(C)NC(c2cc(CC)[nH]n2)=O)c[nH]c2cccc(Cl)c12 69034,Cc1ncc(CC(=O)NC2CC2NC(c2sccc2SC(F)F)=O)s1 69035,c1(NC(C)=O)ccc(F)c(C(=O)NC2CC3CNC(C2)C3)c1 69036,C1(CNC(c2c(C)n[nH]c2C)=O)CCN(C(C2CC2c2nccn2C)=O)CC1C 69037,C1(C(N2C(C)(C)CC(NC(=O)CC3(C(F)F)CC3)C2)=O)CSc2ccccc2O1 69038,N1(C(C(CCC)CC(C)C)=O)CCC(C2(O)CCN(C(=O)CNC(=O)NC)C2)CC1 69039,C1(CC(=O)NCC(=O)NC2CC(n3cnnc3)C2)CCCCC1 69040,c1(C(N2C(C(=O)NCc3ccc(C#C)cc3)CC(F)C2)=O)ccc2c(c1)CCO2 69041,N1(C(C2C(C)CN2C(=O)OC(C)(C)C)=O)CCCCC(C(=O)Nc2ccno2)C1 69042,C1(COC)CC(C)(C)CN1OC(=O)C(C)CCOC1CCC1 69043,C(CCC(C)CC(=O)N1CC(NC(C2(C)CCC2)=O)C2CC2C1)=C(C)C 69044,C1(CNC(c2c(C(C)=O)ccs2)=O)CN(C(=O)C(c2ccccc2Cl)O)CC1C 69045,C1(C(=O)OCC)CN(C(=O)NCC2(c3ccccc3C)CCCC2)CCO1 69046,N1(C(c2c(CSC)ccc(F)c2)=O)CC2(CCCC(NC(=O)OC(C)(C)C)O2)C1 69047,C1(NC(C2(C)CC(C)(C)C2)=O)CCN(C(=O)CC2CC(F)(F)C2)CC1O 69048,CSC1=C(C(=O)NC2CN(C(=O)Cc3nonc3C)CC(C)(C)C2)CCCC1 69049,c1(N2CCC(CC=C)(NC(C3NC(=O)CC3C)=O)C2)nc(Cl)nc(C)c1[N+](=O)[O-] 69050,C1(CCC)COCCN1C(=O)C(CC1CC1)NC(C1CCN(C)CC1)=O 69051,C1(c2ccc(OC)cc2)C(NC(=O)Cc2cccc(SC)c2)CC(=O)N1C 69052,N1(C(CCOC(C)C)=O)CC(CC(=O)NCCc2ncc[nH]2)CC1(C)C 69053,c1(CCCC(=O)NCC2(O)CCN(C(=O)C3CC3)CC2)c[nH]c2ccccc12 69054,C1(NC(c2cn3ccnc3s2)=O)CN(C(C2CC=CC2)=O)C2(CCCOC2)C1 69055,C(=O)(C=C1SCC(=O)N1C)NC12CCCN(C(CC(C)C3CC3)=O)CC1C2 69056,C(=O)(C(C)(C)CC(F)F)N1CCC(N(C(=O)CCCCSCCOC)CC)CC1 69057,C1(NC(C(C)(C)Cc2cccc(Cl)c2)=O)CC2CC(C1)N(C(=O)CCC1CC1)C2 69058,c1(CC)ccc(NCC(=O)N(C2(CC)CCOC2)CC)cc1 69059,c1(C(=O)NC2(CNC(=O)CC3CCC3C)CC(OC)C2)nccc2ccn(C)c12 69060,N1(C(C2(NC(C3(CC(C)=O)CC3)=O)CC(O)C2)=O)CCOC(C2CC2)CC1 69061,C1(O)(C(C)NC(c2cncnc2)=O)CCN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CC1 69062,Cc1cc(=NC2CC(C)N(C(=O)CCCN(C)C)C2)[nH]c(C(C)(C)C)n1 69063,CC1(C)CN(C(C23CC2CCN3C(c2n[nH]c(=N)[nH]2)=O)=O)CCC1O 69064,C1(CC(=O)NCCC2C=CCC2)CCCC1NC(c1cc(CCO)on1)=O 69065,CN(C)S(=O)(=O)N1CCC(C(=O)NC2C=CCN(C(=O)C3=CCCC3)C2)CC1 69066,c1(NC(C2C3CN(C(CCc4c(OC)cccn4)=O)CC32)=O)ccc(Cl)c(F)c1 69067,c1(NC(C2(C)N(c3nc(C)c(Br)cn3)CCC2)=O)ccc2c(c1)OCO2 69068,C(C(C(C)C(C)C)NC(C1(C(F)(F)F)CC(F)(F)C1)=O)NC(CCOCC#C)=O 69069,CCC(C)CCC(=O)NCC(C)C(=O)NC1(CC)CCOCC1 69070,c1(NC(C2(C#N)CCSCC2)=O)cccc2c1C1CCC2O1 69071,C(=O)(C1CCc2ccccc21)N1CCC(C)(CNC(CCC(C)(C)O)=O)CC1 69072,C12(CNC(c3c(COC)scc3)=O)CCCC1CN(C(=O)CCC(C)(C)F)C2 69073,Cc1cccnc1C(=O)NCCC1CCCN(C(=O)CCn2cnnn2)C1 69074,N1(C(CC2OCCN(C(C3C(C)C3C)=O)C2)=O)CC2CCC1C(CO)C2 69075,c1(C(C)NC(C(=C)COCc2ccccc2)=O)ncccc1OC 69076,C1(C(=O)NC2(CN(C)C(C34CC(CC(F)F)(C3)C4)=O)CC2)CCOCC1(C)C 69077,N1(C(C(CC)C)=O)CCC2(CCCN(C(c3ccc(OC)c(NC)c3)=O)C2)C1 69078,Cc1nccc(C(N2CCC(NC(C3CC(C4CC4)C3)=O)C2)=O)c1O 69079,c1(CN2CCC(C(N3CC4(CCC4)C3)=O)C2)c(O)cccc1F 69080,N#CCCCCC(=O)N1CC2C(NC(=O)CCc3ccccc3Br)C2C1 69081,C#CCC(CC(F)F)NC(C1(F)CCN(C(C2(CC(=O)OC)CC2)=O)C1)=O 69082,C1(CNC(CCOCC)=O)CCCN(C(=O)C(C)(C)c2ccccc2)CC1 69083,c1(C(=O)NCC2=CCCN(C(C3(NC(N)=O)CC3)=O)C2)cn2ncccc2n1 69084,c1(C(N2CCC(C(=O)NC3(C)CCCC3(F)F)C2(C)C)=O)cc(C#N)ccc1N 69085,CON=Cc1ccc(C(=O)NCC(C)NC(=O)CC2CCCC23CC3)cc1 69086,c1(OC)ccc(C)cc1C(N1CCC(CO)C(NC(=O)Cc2nocc2C)C1)=O 69087,c1(C(=O)NCCCCC2(NC(C3C(=C)C3)=O)CC2)ccc(=O)n(CCO)c1 69088,Cc1[nH]c2ncnc(N3CCC(C(C)(C)C)(CNC(C4CCOC4)=O)C3)c2c1C 69089,c1(C(C)C(=O)NC2CCC(NC(=O)CSC(C)(C)C)C2)ccc2c(c1)OCO2 69090,c1(C(N2CCC(O)(CNC(Cc3nn(C)c(Cl)c3)=O)C2)=O)cc(N)cnc1Cl 69091,CC1CCCc2nc(C(=O)NCC3(F)CC(NC(=O)C(C)(C)CC4CC4)C3)cn21 69092,C1(C(=O)Nc2ccc(C(F)(F)F)cc2)CC(O)CN(C(c2ccncc2)=O)C1 69093,N1(C(C2(OC)CCSC2)=O)CCC2(NC(c3cccc(=O)o3)=O)CC2C1 69094,C1(C(=O)NC(CC)CN(C(=O)CCC2(C)CC2)C)CCN(c2ncccn2)C1 69095,C1(CC(N2CCC(C(C)NC(=O)CCOC3CC3)C2)=O)CCc2ccccc2C1=O 69096,C(=O)(CCCCCC#N)N1C(C)CC(CCNC(=O)CCC(N)=O)CC1 69097,C(=O)(CCCN=c1nccc[nH]1)N(C)CC1CN(C(C2(N=[N+]=[N-])CC2)=O)CCO1 69098,Cc1ncnc(C(=O)NC2CC(O)(CNC(C3CC3c3cnc[nH]3)=O)C2)c1C 69099,C(C(=O)NCCC(C)C(F)(F)F)(C(C)(C)C)NC(C(OCC)OCC)=O 69100,c1(C(=O)NCC(NOCC)=O)cccnc1CNC(=O)Cc1cccn1C 69101,Cc1cc2ncc(C(N3CCC(C)C(NC(c4nocc4Cl)=O)C3)=O)c(C)n2n1 69102,C(=O)(N1CC(O)CCO1)C1(C)CC(NC(C2CC(=C3CCC3)C2)=O)C1 69103,c1(C(C(=O)NC2C(NC(=O)CCCC3CC3)CCC2)N2CCC2)ccc(Cl)cc1 69104,C(N=c1ccc(C#N)c[nH]1)C1C(NC(COC2C(CC)CCCC2)=O)CCC1 69105,c1(C(N2C(CNC(CC3ON=C(C)C3)=O)COCC2)=O)cc(C)cc2ccoc12 69106,N#Cc1ccc(C(=O)NCCCCCNC(c2cnc(Br)s2)=O)cc1O 69107,c1(OCC(=O)NC(CCCC)CNC(=O)CC2COC(=O)N2)cc(Cl)ccc1C 69108,C(=O)(C(CC1COCCO1)C(F)(F)F)NC1CN(C(C(CC)=CC)=O)CC1SC 69109,c1(Cc2nnnn2CCCF)ccc2c(c1)OCC2.N(CP(C)(C)=O)C(CC)CC 69110,CC1CC=C(C(=O)N2CCCC2CN(c2ncccc2[N+](=O)[O-])C)CC1 69111,c1(NCC)ccc(F)c(C(=O)NC(CNC(=O)CCC2CC2(Cl)Cl)CC)c1 69112,c1(C(=O)NCCNC(=O)CC2CCCC3(CC3)C2)c(F)ccc(C(F)(F)F)c1F 69113,C(C(C(C)C)NC(C1CCC1)=O)OCCSC.C1(=O)CCN1 69114,C1(C(=O)NC(CNC(c2c(OC)cc(C)cn2)=O)C(C)C)CCCC1S(C)(=O)=O 69115,c1(C(=O)NCC2CC(C)N(C(c3ccc(Cl)nc3)=O)C2)nn(C)cc1[N+](=O)[O-] 69116,N1(C(CCSCC)=O)CCN(C(c2cnn(CC)c2)=O)CC1COC 69117,C1(NC(CC)=O)CCC2CN(C(C3(c4cccc(Br)c4)CC3)=O)CCC2C1 69118,c1(C(C)(C)C)cc(Br)cc(Br)c1OC(c1n[nH]cc1C(=O)OC)=O 69119,C=CCCCC(C(=O)NCC(C)(O)CCO)NC(=O)C(C)N(C)C(C)=O 69120,Cc1ccc(SCC(=O)NC2CCN(C(C3CC3C(C)(C)C)=O)C2C)cc1C 69121,c1(C(=O)NC(C(C)C)CNC(c2cncc(C(F)F)c2)=O)cc2ncccc2o1 69122,C1(C(=O)NCC(CC)(C)COC)CN(C(c2csc(Cl)c2)=O)CC(C)(C)C1 69123,N1(CC)CCOC(C(=O)NCCOC2(CO)CN(C(=O)C(CCSC)OC)C2)C1 69124,S(=O)(=O)(c1cnc(NC2CCCSCC2)c(Cl)c1)NC(c1ccoc1)C 69125,c1(C(C)C)c(C(N2CCCC(NC(=O)C=CCF)C2)=O)cnn1CCO 69126,C1(C(N2C(C(C)NC(C3(n4cnnn4)CC3)=O)CCC2)=O)CCCCCC1 69127,CC1(C)CCN(C(=O)CC2CCSC2)C1CC(=O)NC1(C)CC2(CC2)C1 69128,Cc1cc(C)c(NC(=O)C(N2CCCC(NC(=O)CC3(C)CC3)C2)C)c(Cl)c1 69129,C1(NC(C(c2ccc(OC)cc2)=O)=O)CC2CC1CN(C(C1CC1C)=O)C2 69130,N1(C(C(CCOC)C)=O)CCC(CNC(=O)Cc2nc[nH]n2)(OC)CC1 69131,Cc1nc(C)c(C(=O)NC(C2CN(C(c3cocc3C)=O)C2)C)[nH]1 69132,N1(C(c2ccc(Br)s2)C(=O)NCC(=C)C)CC2CN(C)CC2(C)C1 69133,c1(C(N2C(C)(CC(N3CC(F)(CO)C3)=O)CC2)=O)ccc(=N)[nH]c1 69134,c1(Cc2nc(-c3cncc(C(N)=O)c3)on2)cnc(O)nc1O 69135,C(C(CC1CC1)C(=O)NCC1CC=CC1)NC(CC1N(C)CCC1)=O 69136,CC1(CC(=O)OCSC)CN(CCOCCOCCO)C1 69137,C1(C(=O)NCCCC2CCCN2C(=O)CCCc2ccsc2)CC2CCC1CC2 69138,Cc1ccc(Cl)c(NC(=O)C(=O)NCc2ccc(F)c(C)c2)c1 69139,c1(CC)nc2sc(C)cn2c1C(=O)NCC1(O)CCCCCC1 69140,N1(CC(n2cc(-c3ccc4c(c3)OCO4)nn2)C)CC(CO)Oc2ccccc21 69141,N#Cc1cccc(F)c1CC(N1CC2CC(NC(=O)C#CC3CCC3)C1C2)=O 69142,C1(C(N2CCC(C(C)NC(c3cnc(C(F)(F)F)s3)=O)C2)=O)CCS(=O)(=O)N1 69143,C1(CC)CN(C(=O)CCOCC2CC2)CCC1NC(=O)CC1CCC=CCC1 69144,Cc1cc(C(N2CCC(F)(C(=O)Nc3ccc(F)c(I)c3)CC2)=O)cnc1Cl 69145,N1(C(C2CN(CC)C(=O)C2)=O)CC(C(=O)NCC(CSC)OC)CC12CCC2 69146,N1(C(C)=O)CC2(CC(NC(c3cnc(N4CCOCC4)nc3)=O)C2)C1 69147,c1(C(N2CCCC(CCNC(C3CC(=C4CC4)C3)=O)C2)=O)cc(F)c(O)c(F)c1 69148,C1(C(=O)NCC=CCSC)CCCCC1.c1(NC(=O)COC)cccnc1 69149,C(C)(C)(C(=O)NCCC1(CNC(C2CSCCS2)=O)CC1)OCCC 69150,C(C)(C(=O)N1CC(OC2CCOCC2)C1)(C(C)C)SC 69151,c1(C(C)(C)C)nocc1C(=O)NC1COCC1NC(=O)C(F)CC1CCCC1 69152,c1(OC)ccc(Cl)cc1COC(N1CC(OC(c2cc(C3CCC3)on2)=O)C1)=O 69153,Cc1nc2ccccc2nc1NC(c1ccc(CN2CCOC(C)(C)C2)cc1)=O 69154,C(=O)(C(C)CC(F)(F)F)NC1(CNC(c2ccnc(CO)c2)=O)CC(OC)C1 69155,c1(C(C)=O)cnc(NC(=O)CC2CN(C(=O)C3=COCCC3)CCO2)nc1C 69156,N1(C(C2CC(=O)C2)=O)CC(N=c2ccn3ccnc3[nH]2)CC2(CCC2)C1 69157,C1(c2nnnn2CCO)(CCO)CCCC(C(F)(F)F)C1.CC(C)(C)CCCN 69158,c1(C(=O)NC2C(CNC(c3ncc(NC)nc3)=O)C2)ccc(F)c(Cl)c1F 69159,C1(C(=O)OC(C)(C)C)CCCC(OCC(N2CCCC(CC#N)C2)=O)C1 69160,C(=O)(CCC(C)(C)C#N)N(c1ccc(C)cc1)CC(=O)NC(COC)C 69161,C(CC1=CCOCC1)NC(C1C(NC(=O)CCOC2CCCC2)CC1)=O 69162,Cc1ccn2cc(C(=O)NC3CN(C(C4CCC(N=[N+]=[N-])C4)=O)CC3(C)C)nc2c1 69163,N1(C(CC2(C)CC2)=O)CC2CCCC(C1)N2C(=O)CC1CCCCCC1(F)F 69164,CC1CS(=O)(=O)CC(C)N1C(C1SCCS1)=O 69165,C1(CNC(CCC=C)=O)CCC2(CCC2)C1NC(=O)CCN1CCOC1=O 69166,C(=O)(C1=CCOCC1)NCc1cc(C(N(C2CCCC2(F)F)C)=O)on1 69167,c1(C(N2CCCC(OCC3CC3)C2)C(=O)NC2CCC2)ncccc1F 69168,C1(CC)CN(c2nnc(CSCCO)n2CC(=O)NC)CC(C)O1 69169,c1(CNC2CN(C(c3ccc(F)c(F)c3)=O)CC(F)C2)cc(Cl)c2cn[nH]c2c1 69170,c1(OCCC(=O)NCCC2CC(NC(C3CCSCC3)=O)C2)c(F)cccc1Cl 69171,c1(CC(C)C)ccccc1C(=O)NC(C)(C)CNC(=O)CCN1CCNC(=O)C1 69172,c1(C(=O)NC2CCCN(C(c3ccc(O)cc3)=O)C2)csc2ccc(Cl)cc12 69173,N(C(=NCCn1cccn1)NCc1ncccc1O)CC1N(CC)CCC1 69174,c1(OC(C)C)c(F)cc(-c2nc(NC(=O)CNc3nccs3)cs2)cc1F 69175,c1(C(=O)NCCN(CCC)C(N)=O)cc(F)c(F)cc1NC(=O)Cc1cnns1 69176,N1(S(Cc2ccc(C)c(F)c2)(=O)=O)CCN2CCOCC2C1 69177,C(=O)(C(=O)CC(C)CC)NCC1(CC(=O)N(C2CC(=C)C2)C)CC1 69178,Cn1c(C(N2CCC(O)(CNC(=O)CC3CCCOC3)CC2)=O)cc2sccc12 69179,N1(C(=O)C=Cc2ncc[nH]2)CCC2OCCN(C(C3CCC(F)CC3)=O)C2C1 69180,c1(C(=O)NC2CCN(C(C(C)NC(=O)C3CC3)=O)C2)ccnc2ccc(Cl)cc12 69181,C(=O)(C(CC(C)C)C(N)=O)N1CCCC(CN(C(C(CCC(C)C)F)=O)C)CC1 69182,N(C1CCCc2n[nH]cc21)C(C(C)(N(C(=O)CCn1cnc(=N)[nH]1)C)C1CC1)=O 69183,c1(C(=O)NCC(CO)NC(c2cnc(Cl)s2)=O)cccc2nccnc12 69184,N1(C(c2ccc(Cl)s2)=O)CC(CNC(C23COCC2C3)=O)C2(CCC2)C1 69185,Cc1nc(-c2cn(CC(C3CN(C(C4(C)CC4F)=O)C3)F)nn2)sc1C 69186,C1(NC(c2[nH]c(=N)sc2)=O)CCCC2CN(C(C3CCCC(F)(F)CC3)=O)CC12 69187,O=C(N1CC(n2cc(C3CCCCO3)nn2)CO1)c1cncc(C2CC2)c1 69188,Cc1nc(O)ccc1C(N1CCC(C(=O)NCCc2c(C)n[nH]c2C)C1)=O 69189,c1(CC=C)ccccc1C(=O)NCCCCCNC(=O)C(COC)N(C)C 69190,C=CCC(CNC(=O)CN(C)C(N)=O)C(=O)NCc1nnn(C)c1C 69191,C1(CN(C(c2ccc(C(F)F)s2)C(=O)NCCC2CC2)C(CC)C)CCCCC1 69192,Cc1cc(C(=O)NC23CC(C2)N(C(c2cccnc2SC(F)F)=O)C3)cc(Cl)c1 69193,C1(NC(c2n(C)c(S)nn2)=O)CCCC(C(N2CCCC2(C)C2CC2)=O)CC1 69194,C1(C(N2CC(NC(=O)C(C)(C)C#N)CC(C)(C)C2)=O)Cc2cc(Br)ccc2O1 69195,N1(C(CSC)=O)CC(NC(=O)CSc2cccc(Br)c2)CCC1C 69196,c12ccc(cc1)NCCCCc1cn-2nn1.c1(C(=O)OC)c[nH]c(C(=O)NC)c1 69197,CC(C)(C)C(C(=O)NCc1ncoc1CCNC(c1n[nH]cc1Cl)=O)NC(N)=O 69198,N1(C(c2c(C)ccnc2C)=O)CC2CCC(C1)C(NC(c1ccoc1C)=O)C2 69199,N1(C(C(c2c(C)cccn2)(F)F)=O)CC2(CCC2NC(C2CNC(=O)C2)=O)C1 69200,CCC(CC)C(=O)NC(C)(CNC(c1cccc(C(=O)N(C)C)c1)=O)C(C)C 69201,C1(CC)CN(C)CCCN1C(=O)COC1(C)CN(C(=O)CC23CCCC2C3)C1 69202,C1(N(C(C2CCCOC2)C(=O)NC)C)CCC(OC)CC1 69203,C(C)(C)(CCCC(=O)NCCCC1CCCC1O)NC(c1c(C)cc(O)nc1)=O 69204,C(=O)(C(O)CC(C)C)NC(CCN(C(c1cc(OC)ns1)=O)C)C(C)C 69205,C1(NC(c2cnn(C(C)C)n2)=O)CC(C(=O)NCc2snnc2C)C12CCC2 69206,N1(Cc2c(C(=O)OCC)n[nH]c2)CC2CN(C(c3cc(B(O)O)co3)=O)CC12 69207,Cc1ccccc1C(C)C(=O)NCC(C)CN(C(=O)C(C1CCC1)C1CCC1)C 69208,Cc1cc(-n2cccn2)nc(=NCC2C(C)CCCN2C(=O)C(C)CN(C)C)[nH]1 69209,c1(C(N(CC(C)NC(=O)CCCC#N)C)=O)ccc(-n2cccn2)cc1 69210,c1(N2CCC(Br)=C(C)C2)ccc(S(=O)(=O)NCC2Cc3ccccc3CO2)cc1Cl 69211,c1(C(=O)NC(CC(C)NC(=O)CC2CCN(C)C2=O)C)cc(N)c(F)c(F)c1F 69212,c1(OC)cc(OC)c(C(=O)NCC2CCC2NC(c2nncs2)=O)cc1OC 69213,Cc1nc(-c2ccc(COc3ccccc3)cc2)ccc1C(=O)NC1CNC1 69214,N1(C(C)=O)CC(c2nnnn2C(C)C)(NCCC2CCCC2O)C1 69215,C(=O)(C(C)S(=O)(=O)C(C)C)NCC(C)(C1CCC1)NC(C1CCC(CC)O1)=O 69216,c1(CC)c(Cl)nc[nH]c1=NCC(O)CNC(c1cc(O)c(F)c(F)c1)=O 69217,c1(C(N(C(CNC(c2ccc(N)cc2Cl)=O)C2CC2)C)=O)ccn2nnnc2c1 69218,C#CC(C(C)OC)NC(C1(C(C)NC(C2CC(CC)C2)=O)CC1)=O 69219,CC(CCC#N)(c1nnnn1Cc1ccccc1)NCCc1cccnc1 69220,Cc1nn(CC(=O)NC(C)C(C)NC(=O)C(CO)c2ccccc2)cc1Cl 69221,C1(OC)CN(C(c2sccc2I)C(=O)NC2CCOC2)C2(CCC2)C1 69222,c1(C(N2CC3CC(C2)N3C(c2cnc(Cl)nc2)=O)=O)ccc2nc(Br)sc2c1 69223,N1(C(C23OCC(C(C)C)(C2)C3)=O)CCC(C)(NC(=O)CCS(N)(=O)=O)CC1 69224,Cc1cc(C)c(C(=O)NCC2C(C)CCN2C(=O)CCc2csc(=N)[nH]2)o1 69225,c1(C(N2CC(SC)C(NC(=O)C=CSC)C2)=O)ccn(CC(F)(F)F)c(=O)c1 69226,C1(O)(CN(C)C(c2ccoc2)=O)CCN(C(C2CCC(c3ccccc3)C2)=O)C1 69227,C(C)(C(CCc1cn[nH]c1)NC(c1[nH]c(O)nc1C)=O)NC(CSC)=O 69228,C(N=c1[nH]c(N(CC(N)=O)C)nc2c1SCC2)C1CCN(S(C(C)C#N)(=O)=O)C1 69229,N1(C(c2nnc(-c3cc4c(s3)CCCC4)o2)C)CC2OCCN(C)C2C1 69230,N1(C(C2C3CC(=O)CC32)=O)CC2C=CC1C(C(=O)NCC1(O)CCOC1)C2 69231,N1(C(C(CO)NC(C(C)C)=O)=O)CCC(NC(=O)CCc2c[nH]c(=N)[nH]2)C1C 69232,C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC(C(=O)NC(C2C(CC)C2)C)C1 69233,C1(C(N(CCNC(CC2(C#N)CC2)=O)CCOCCO)=O)CC12CCCC2 69234,C(C)(CCC(=O)NC(CNC(=O)C(C)(C)c1cnc[nH]1)CO)OC 69235,C1(C(=O)NC(C#C)CC2CCC2)CC2CC2N1C(=O)C(C)NC=O 69236,N1(C(COCc2cc(C)on2)=O)CCN(C)CC1CNC(C1(C(N)=O)CC1)=O 69237,n1(CC(=O)OC)nc2c(c1NC(=O)C(N1CC(CO)OC(C)C1)=O)CCC2 69238,N1(C(C=CCCC=C(C)C)=O)CCC(NC(=O)C=Cc2cc[nH]n2)C(C)C1 69239,CN1CC(F)CC1C(N1CCC(NC(=O)CCCc2cncs2)C1)=O 69240,C1(CC(=O)NC2CN(C(c3cc(F)c[nH]3)=O)CC2CC2CC2)CCCS1(=O)=O 69241,C1(C)(C(N2CC(C)(CSC)C2)=O)CCN(C(=O)C(O)C(C)(C)C)CC1 69242,CC(C)C(C(=O)NCC(C)N(C(=O)C(F)C1CCOC1)C)n1ncc(N)n1 69243,C1(N(CCCC(=O)N(C(C)C)CC)C)CCN(C(=O)OC(C)(C)C)C1C(C)(C)C 69244,C(=O)(C(C)(O)C(F)(F)F)NCCC(C)NC(=O)C(O)CC1CCOCC1 69245,c1(C(N2CCC(NC(C(COC)C)=O)C23CC3)=O)ccc2cccc(C)c2n1 69246,CCS(=O)CC(=O)NCCC1(C)CN(C(=O)COCCN(C)C)C1 69247,C1(NC(CCN2C(C)CCCC2)=O)CC(F)CN(C(=O)CC2CC3(CCC3)C2)C1 69248,c1(-c2scc(C(=O)NNC(c3cccc4[nH]ccc34)=O)n2)cccc2c1OC(F)(F)O2 69249,c1(C(=O)NC(CNC(CC2(C=C)CCOCC2)=O)CO)ccc(F)c(C)c1F 69250,C12(C(C(C)N(C)CC3(c4ccc(Cl)cc4)CC3)=O)CC3CC(CC(C3)C1)C2 69251,C1(COCC)(Nc2c(C(=O)NC)n[nH]c2)CCOCC1.C12(CCC1)C(=O)NCC2 69252,C1(CNC(c2c(CC)cns2)=O)CC(C)(C)CN1C(c1ccc(F)cc1N)=O 69253,c1(C(C(=O)OC(C)(C)C)NC(C(=O)NC(C(CC)C)=O)=O)cccc(F)c1 69254,c1(CC)nc2sc(C)cn2c1C(=O)NC1CCC1NC(c1ccoc1CC)=O 69255,C1(NC(CC(C)(O)c2ccccc2)=O)CC2(C1)CC2N=c1[nH]nc(C#N)s1 69256,c1(CNC(CC(COC)(C)C)=O)nc2c(s1)CN(C(c1ccnnc1)=O)CC2 69257,c1(C(=O)NC2CN(C(C3C(OCC)C3C)=O)C2)ncccn1 69258,c1(NC(=O)CC2CCC(NC(c3nc[nH]n3)=O)CC2)cc(Br)nc(Br)c1 69259,N1(C(CCc2ccc(C)nc2)=O)CC2(C1)CN(C(C13CC1COC3(C)C)=O)C2 69260,N#Cc1ccccc1C(=O)NCCc1cc(C(N2CCC(F)(F)C2)=O)no1 69261,C(=O)(CCCN=C(NCC(C)(C)C)N1CC2CCN(C)C2C1)N(C)C 69262,C(=O)(CCC1CCc2ccccc21)N1CCCC(C)(CN=c2[nH]nc(CO)s2)C1 69263,C(=O)(CC(C)C(C)C)N1CCCC(CN(C(CCC(=O)NCC)=O)CC)C1 69264,N1(C(C2OCCN(C)C2)=O)CC2CC1CN2C(=O)COCCc1ccccc1 69265,c1(CC)c(C(=O)N(C)CCOCCNC(C2CCCC2C(C)C)=O)cnn1C 69266,C(=O)(C(CC)C(C)C)NC(CC=C)CNC(c1cnn(C)c1COC)=O 69267,c1(CC)ccc(C(=O)NC2COCCC2NC(=O)Cc2ccc(C)cc2)c(O)c1 69268,c1(C(=O)NCC(CCNC(c2nnn(C)c2N)=O)O)ncc(F)cc1F 69269,C12(C(N3CCC(C)(C)C3)=O)CCC(CN(C(=O)CC3CCCO3)C1)C2 69270,N1(C2CC(NCC(N3CC(C4CC4)C3C3CC3)=O)C2)C(=O)c2ccccc2C1=O 69271,Cc1ccc(CC(=O)NC2CCC(NC(C3CCC4C3C4(F)F)=O)CC2)cc1Cl 69272,N1(C(C(CC)C#N)=O)CC2CC1CN2N(c1ccnc(O)c1Br)C(=O)C(F)(F)F 69273,c1(OC)cnnc(C(=O)N(CCCOCCNC(C2(N=[N+]=[N-])CC2)=O)C)c1 69274,C1(CNC(c2scc(OC)c2)=O)CCC2CN(C(=O)CCc3cc(C)[nH]n3)CC12 69275,c1(C(=O)NC(C)(C)CNC(C2CCCCS2(=O)=O)=O)cc(Cl)cc2ccncc12 69276,c1(OC)c(CNC(=O)Cc2ccc(-n3cnnn3)cc2)cccc1Cl 69277,CC(C)C(F)C(=O)NCC1(C(=O)NC(C)Cc2ccccn2)CC2(CC2)C1 69278,CC1CCC(NC(C2(Oc3ccccc3)CC2)=O)CN1C(C1C(C)(C)C1(C)C)=O 69279,C12(C(=O)NCC=C(C)C)CC(CO1)N(C(c1cccc[n+]1[O-])=O)C2 69280,c1(C(N2C3CCC(CNC(c4c(OC)n[nH]c4)=O)(C3)C2)=O)c(O)nnc(C)c1C 69281,C1(NC(Cc2ccc(C(C)=O)s2)=O)CC2CN(C(C3C=C3C)=O)CC12 69282,C1(C)(NC(C(C)O)=O)CC(NC(c2[nH]ncc2C2CCC2)=O)C1 69283,c1(C(C)NCCN(CC(F)(F)F)CCO)c[nH]c2ncccc12 69284,C(C(C)C(C)C(=O)NCCOC1CCN(C(C2CC3(CSC3)C2)=O)C1)OC 69285,N1(C(c2n(CC)cc(Cl)c2)=O)CCC(CCNC(c2n[nH]c(C)n2)=O)C(F)(F)C1 69286,Cc1nn(C2CC2)cc1CNC(c1nnnn1CCOC1CCCC1)CC1CC1 69287,Cc1cc(C(N2CCC(C(N)=O)(Nc3ncccc3C#N)CC2)=O)c(C)cn1 69288,N1(C(C(C)CC2CCCC2)=O)CCC(CC(N)=O)(NC(c2cnn[nH]2)=O)CC1 69289,c1(C(=O)NCC=CCNC(C2CCC2F)=O)ccc(-c2nc(=O)o[nH]2)cc1 69290,c1(C(=O)NCCS(C)(=O)=O)cc(C2=CCSCC2)c2cc[nH]c2c1 69291,CC1(C#CC(=O)N2C(C(=O)NC3CCN4CCCC34)CC3CCCC23)COC1 69292,Cc1ncc(C(=O)NCC2(F)CN(C(C3C4CC4C4CC34)=O)C2)c(C2CC2)n1 69293,CCCCCCC(=O)NC(C)CCN(C(=O)C(C)OCCN(C)C)C 69294,Cc1cncc(C(N2CCC(NC(C34CCCC3C4(F)F)=O)C(O)C2)=O)c1Cl 69295,C1(NC(=NCC=C)NCCCCN2CCCC2)CCc2cc(OC)ccc2C1 69296,C1(NC(C(CC)F)=O)C2CC1CN(C(c1cccc(-n3nc(C)cc3C)c1)=O)C2 69297,N1(C(C(CC)=Cc2cccnc2)C(=O)NCC(C)C)CC(C)(C)OC2COCC12 69298,N1(C(c2cnc(COC)s2)=O)CCC(NC(=O)CC2CC(F)(F)C2)C2(CCC2)C1 69299,c1(NC(c2n(CCC(=O)OCC)nnn2)C2CCC2)ccc2nc(C)ccc2c1 69300,c1(C(=O)NCC2(O)CC(NC(C=CC(C)(C)SC)=O)C2)cc2n(n1)CCC2 69301,c1(CC(=O)N2CC2)cc(Cl)ccc1Cl.N1(CC)CCC1C(=O)OCCSC 69302,C1(C(=O)NC(CNC(C(C2CC(F)(F)C2)OC)=O)(C)C)CCC2(CCC2)CO1 69303,C1(OCC(=O)NCC2CN(C(C3CC(O)C3)=O)C2)CCCCCC1 69304,c1(OC)ccc(SCC(N2CC(CO)(NC(=O)CCNC(N)=O)C2)=O)cc1 69305,n1(CC)nc(C2CC2)cc1C(=O)NCC12CC1CN(C(C1(O)CCSCC1)=O)C2 69306,N1(C(C2N(C(=O)OC)CSC2)=O)CC2CCC2(C(=O)NCc2cc(F)cc(F)c2)C1 69307,c1(C(N(C2CN(C(=O)CC(F)(F)c3ccccc3)C2)C)=O)nccc2ccsc12 69308,CC1(C)CCC(C(N2CC(NC(c3cnc(O)c(F)c3)=O)CC(F)C2)=O)CO1 69309,C1(C(=O)OC)CC1C(=O)NCC=CC(=O)NCC1CC1Cl 69310,C(C(CC(C)C)C(=O)N1CC(C(C)NC(=O)C(C)(C)C(C)O)C1)OC 69311,C1(NC(c2ccc(C(F)F)cc2)=O)CCCCC1N(C(C1(CF)CC1)=O)C1CC1 69312,Cc1c(C(=O)NC2CC3CC(NC(=O)CC4(C)CCC4)CC23)nn(C)c1N 69313,C1(NC(CN(C)CC)=O)CCC(C)(CNC(c2ccnc(C3CC3)c2)=O)C1 69314,C(=O)(C1=CCSC1)NC1C(CC(=O)Nc2ccccc2)C(O)C1 69315,C(CCC)(C(=O)N1CC2C(CN(C)C)C2C1)NC(CC1CC(OCC)C1)=O 69316,Cc1c(C(=O)NC2CCCN(C(=O)CSC3CC3)CC2)cncc1F 69317,c1(C(=O)NC2CN(C(c3cccc(CC)c3O)=O)C2)ccc2cc(C)ccc2c1 69318,CC1CCN(C(=O)CCNC(=O)C2CC2)C1CNC(=O)C(=O)NC1CCCC1 69319,N1(C(C(=O)NC2CC2)c2cnc[nH]2)CCC2(CCCCC2)CC1 69320,N1(C(C=CC(=O)OCC)=O)CC2CCC1C(NC(=O)CC1CC(SC)C1)C2 69321,C(=O)(CCC(C)(C)[N+](=O)[O-])N(CCCC(=O)N(C(C)CO)C)C 69322,C1(COC)(CNC(=O)Cc2coc(C)n2)CCN(C(=O)C(C)N=[N+]=[N-])C1 69323,N1(C(CC(C)(C)C)C(=O)NCc2cccs2)CCn2c(Br)cnc2C1 69324,c1(C(=O)NCC2(Oc3scc(CNC(=O)COC4CC4)n3)CC2)ccccn1 69325,C(=O)(C1=C(CC)OCCC1)N1CC(C(N2C(CC(=O)OCC)CCC2)=O)NCC1 69326,C1(N(C(=O)CC(F)(F)F)C)CCCN(C(=O)CNc2ncccn2)CC1 69327,N1(C(Cn2c(C)ccc2C)=O)CCN2CCN(C(=O)C(O)C(C)(C)C)CC2C1 69328,C1(C(=O)NCCC(C)NC(C23COC(C2)C3)=O)CCCCO1 69329,Cc1nc2cc(NC(C3CC34CC4(F)F)=O)ccc2n1C(CO)CO 69330,C1(NC(Cc2ccc(C)s2)=O)C=CCN(C(c2ccnn2C(C)C)=O)C1 69331,C1(CNC(CC(C(C)C)C)=O)CC2CCC1N(C(=O)CC1C=CCCC1)C2 69332,c1(CN(c2ncc(OCC)cn2)C23CCC(N)(CC2)C3)cc(F)ccc1C 69333,c1(C(N2CC3(N(C(C4CCC(C)(C)OC4)=O)CC3)C2)=O)cccc2nn[nH]c12 69334,C=C(C)CCCC(=O)N(C(C)CNC(=O)CCCC(=C)C)C 69335,CCC(CC(=O)N(CCCC(=O)NCC1C=CCCC1)C)CC(C)C 69336,C=C(C)CC(C)C(=O)NCC1CCN1C(c1cc(F)cnc1OC)=O 69337,C1(C(=O)NCC(C)(C)NC(c2cnc(Cl)cc2N)=O)CCc2ncncc2C1 69338,C1(NC(=O)NCCC(COC)C)CC(=O)CCO1 69339,c1(C(=O)NCC(CC)NC(C23CCCC2C3(F)F)=O)ccc(OC)c2ccsc12 69340,c1(C(N2C(C)CC(CNC(c3n(CC)nnc3)=O)C2)=O)occ2c1CCC2 69341,CC(CC(C)(F)F)C(=O)NCC(C)(C)Cn1cc(C(O)C(C)(C)C)nn1 69342,C(=O)(CC(C)(F)F)N1CCC(n2cc(CNC(CN(c3ncccn3)C)=O)nn2)C1 69343,CC(=O)CCCC(C)C(=O)N1CC2CCCC2C1C(=O)NCC1CC1 69344,c1(C(=O)NCCC2CCN(C(Cc3scc(C)c3)=O)C2)cccc(C(N)=O)c1 69345,N1(C(Cc2cc(C)sc2C)=O)CCCC(N(C)C(C2CCCC(C#N)C2)=O)CC1 69346,C(C)(CCN=c1[nH]cc(C(=O)OC)cc1C)NC(CCCC(=O)NC)=O 69347,N1(C(C(C)NC(CC)=O)=O)CC=CCC1C(N1CCN(C(C)C)CC1)=O 69348,c1(NC(C(=O)N(CC(C)C)Cc2ccccn2)=O)ccc(C2CCC(=O)N2)cc1 69349,C(=O)(C(O)C(C)(C)C)N(CCN(C(c1sc(CCC)c(CC)c1)=O)C(C)C)C 69350,c1(CC(=O)NCC(CO)NC(CCc2ncc(C)[nH]2)=O)ccnc(Cl)c1F 69351,C1(NC(c2nnnn2CC(F)F)(C)C2COC2)CCN(C(=O)C2CC2)C1 69352,C1(NC(C(COCC)CC)=O)CCN(C(=O)CCCN(C)C)CC1(C)C 69353,N1(C(COCCOC)=O)CCOC2(C1)CN(C(C1(C)CCCNS1(=O)=O)=O)C2 69354,N1(CCNC(C2(C)C(C)C2)=O)CCC(NC(C2CCC2(F)F)=O)CC1 69355,C(=O)(C1=NN(C)C(=O)CC1)N1CCC(NC(C2(C(=O)NC)CC2)=O)C(CO)CC1 69356,C1(C(=O)NC(c2ncccn2)(C)C)CCC2(CC2)N1C(=O)CCC1CCC1 69357,C1(NC(C(C(CC)C)OC)=O)CCCC12CN(C(c1ccsc1SC)=O)C2 69358,CC(C)C(C)C(=O)N1CC2CC2(NC(c2cc(-c3ccccc3F)on2)=O)C1 69359,CCC(C)(C)C(=O)NCC1(CC(=O)OC)CC1.C12CC(C1)N(C)C2=O 69360,C(=O)(C#CC1CCC1)NCC(C)CN(C)C(C1C2CCCC12)=O 69361,CC1CC2(CCN(C(=O)C3=CC4CCCC34)CC2)CN1.C(C)C(=O)NC1CCCO1 69362,n1(SCC)nncc1CN1CCC(N(C)C(=O)OC(C)(C)C)C1 69363,c1(C(N2CCN(CC(N)=O)CC2)C(=O)NCCCSCC)ccc(C)c(F)c1 69364,C1(C(N2CCC(F)(CNC(C(C)(C)SC)=O)C2)=O)CCC2(CCCC2)C1 69365,N1(C(C(=O)NC2CCN(Cc3cn(C=C)nc3)CC2)=O)CCCCC(C)C1 69366,C#CC1(OCC(=O)NCCNC(=O)C(c2cnn(C)c2)O)COC1 69367,C1(NC(=O)Cc2cccc(Cl)c2)CC2CCC(C1)N2C(C12COC(C1)C2)=O 69368,CCCCCC(O)CC(=O)N(C(CC(F)F)C(=O)N(CC1=CCSC1)C)C 69369,c1(NCC2(C)N=C(C)SC2)ccc(S(=O)(=O)N(CC(C)(C)CO)C)c(Cl)c1 69370,C1(CC=C)(NC(=O)CCCc2cccs2)CCN(C(=O)CCOCCOC)C1 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69457,C(=O)(C(F)(F)C(F)(F)C(F)F)N1CCC(N(C(C2CC23CCOCC3)=O)CC)C1 69458,C1(CNC(CCC(N)=O)=O)CCC2(CCC2)C1NC(=O)CC1=NNC(=O)C1 69459,Cc1cc(=NC(C)CNC(c2ncncc2Cl)=O)[nH]cn1 69460,O=C(C1=CCCN(Cc2c[nH]c3ccccc23)C1)N(c1ccc(F)cc1)CCO 69461,C1(NC(C(=O)N(CCCN2CCCC2)CC)=O)C[Si](C)(C)CC1O 69462,N1(C(CCSCCC)=O)CC(NC(C2CCCC(=O)C2)=O)C(C)C1 69463,CCCCC(C)CCC(=O)NC(C)C(C)(C)NC(=O)Cc1ccc(O)c(C)c1 69464,C1(OC(C)(C)C)(CON2CCOCC2c2nc[nH]n2)CCS(=O)(=O)C1 69465,C(=O)(CC1COc2cc(O)ccc21)N(CC(C)NC(c1ccc(C)nc1)=O)C 69466,N1(C(COCCCOC)=O)CCC(C)C(NC(=O)C(F)=C(C)C)C1 69467,c1(C(N2C(CN(C(C(CC=C)C)=O)CC)CCC2)=O)ccc(NC(C)=O)cc1Cl 69468,CCCC(C(=O)OC)C(=O)N1CC(C)CC1C(=O)NCCCC(C)C 69469,Cc1ccc(NC(=O)C=C2CCN(Cc3c(Br)cnn3C)CC2)c([N+](=O)[O-])c1 69470,c1(C(=O)OCc2onc(C(C)(F)F)n2)cc2cc(Cl)ccc2[nH]1 69471,c1(NCCC=CC=C)cc(=NC(C)c2ccn(C)n2)[nH]c(COCC)n1 69472,Cc1cc(C(=O)NC2CC2NC(=O)C2=C(Cl)CCC2)cc(O)n1 69473,N1(C(c2c(C)onc2)=O)CCCC(C(C)NC(=O)CC2(c3ccon3)CCC2)C1 69474,c1(C(N2CC(CCC)N(C(c3cnnn3C)=O)CC2)=O)ccn2cccc2c1 69475,C=C1CCN(C(c2nc(C)sc2C)=O)C(C(N2CCCC(C(C)C)CC2)=O)C1 69476,C1(C(=O)NCC(CNC(=O)C(C2CCOCC2)C)CO)(CC)CCCC1 69477,CCC(CNC(c1ccccc1Cl)=O)(CC)C(=O)NCCS(=O)C(C)(C)C 69478,C(C(CC(C)C)NC(c1csc(F)c1)=O)NC(c1n(CCC)ccc1)=O 69479,CC(F)(F)CCC(=O)N1C2CCC1C(CNC(c1ccnn1CC1CCC1)=O)C2 69480,N1(C(CCC2N(C(c3c(CC)cco3)=O)CCC2)=O)CCC(C)C2(CCC2)C1 69481,c1(CN(CCCCOC)CCC)csc(-c2cnn(C)c2)n1 69482,CC1CN(C(=O)CC(O)C2CCCC2)CCC1NC(c1cn(C)ccc1=O)=O 69483,N1(C(CC2CC(=C)C2)=O)CCN(C(=O)Cc2ccc(O)cc2)C2CCCCC12 69484,C1(NC(CN(CC)CC)=O)CC2(C1)CC(C(=O)NC1CCC3CCC13)C2 69485,N1(C(C(C)OC)=O)CCC(F)(F)C(N=c2nc(C)nc3[nH][nH]cc2-3)C1 69486,N1(C(CNC(=O)OC)=O)CC2CCC2(CC(=O)NC2CC(=C3CC3)C2)C1 69487,C1(O)(CCNC(COCc2nnc(C)s2)=O)CCN(C(c2cnc(O)o2)=O)C1 69488,Cc1cc(C(N2C(C(N3CCC(F)(F)C3)=O)CC3CC23)=O)c(C)cc1Br 69489,C(=O)(C1CCCc2scnc21)N1C(C)(C)CC(NC(C2CCC(C)CC2)=O)C1 69490,C1(N(C)C(c2cc(C(F)F)no2)=O)CCC(NC(=O)C(C)(C)C#N)CC1 69491,CC1CC(C(=O)Nc2c[nH]nc2Br)N(C(c2cncc(Br)c2)=O)C1 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69510,S(=O)(=O)(c1c[nH]c(C(=O)NC2CN(C(=O)C#CC3(C)CC3)CC2C2CC2)c1)NC 69511,N1(C(CC=C=C)=O)CCCC(NC(c2nc(C)n(C3CC3)c2C)=O)C1C 69512,C(CCC(=O)NCCC1(NC(=O)CCF)CCCC1)=CC 69513,S(=O)(=O)(c1cnc(NCC2CCC2(F)F)c(Cl)c1)NCC(C(CC)CC)O 69514,N1(C(COS(CC)(=O)=O)=O)CC(NC(c2cccc(OC)c2OC)=O)C2(CC2)C1 69515,CC1CCCCC1CNC(=O)CC(c1cccc(Br)c1)C 69516,Cc1ccc(F)c(C(=O)NCc2cccc(CNC(c3cn(C)cn3)=O)c2)c1F 69517,C(=O)(C(CNC(C1(CO)COC1)=O)C(C)(C)C)N(CCC)CC 69518,CC1CCC(NC(=O)Cn2cnc(=N)[nH]2)CN1C(=O)CC1(CO)CC1 69519,N1(C(CNC(=O)NC)=O)CCN(C(c2cccc(OC(C)=O)n2)=O)C(C)CC1C 69520,CC1(C(=O)NCC2(O)CCN(C(=O)CCCn3cccc3)C2)CCCNS1(=O)=O 69521,N1(C(c2cn(CCC)nc2)=O)CCOC(CNC(=O)Cn2[nH]cnc2=N)C1 69522,c1(C(=O)NC2(C)CCC(NC(C(C)(C)OC)=O)CC2)cc(C)c(F)cc1N 69523,c1(C(=O)NCC2N(C(C3CCN(C)C3)=O)CCOC2)cncc2c(F)cccc12 69524,c1(C(=O)NC2(C)CN(C(C(CCC)(C)C)=O)C2)n[nH]c2c(C)cccc12 69525,Cc1cccc(C(=O)N(C(C)CNC(c2nn(C)cc2Br)=O)C)c1 69526,C(=O)(CC1=CCCCC1)NCC(C)CNC(c1conc1C(F)(F)F)=O 69527,c1(C(=O)NCCCCC(C)NC(=O)CSC(F)F)ccn2nccc2c1 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69702,N1(C(c2nc(OCC)oc2)=O)CCC2(CC1)CC(NC(=O)CCC(N)=O)CCO2 69703,C1(C(C(=O)NCCNC(Cc2ccc(C(C)=O)s2)=O)C)CCCCCC1 69704,CC1(CCNC(C2(C)CCCCC2)=O)CCN(C(=O)C=C2CCCCC2)C1 69705,Cc1cc(Br)cc(S(=O)(=O)NCCC2(C)NC(=O)NC2=O)c1 69706,c1(C(C(=O)NC2CCOCC2)N(C(CCO)C(F)F)CC)cc(OC)ccc1Br 69707,c1(NC(=O)OCC)ccc(NC(C2(C(C)(C)O)CCOC2)=O)cc1 69708,c1(OCC)cc(C(=O)NCC23CC(NC(c4cccnc4)=O)(CO2)C3)ccn1 69709,C1(NC(C(=O)N(CC(C)CN(CC)CC)CC)=O)CC[Si](C)(C)C1 69710,C1(OCC)(CNC(=O)CC2COC(=O)N2)CN(C(=O)CN2CCSCC2)C1 69711,C1(NC(c2cn(CCOC)nc2C)=O)CN(C(C2CC3C=CC2C3)=O)CC2CC12 69712,CCC(C)(CNC(C1CC1(F)Cl)=O)C(=O)N(CC(C)(C)OC)C 69713,N12CCCC(C1)C2=O.C1(C(C)=O)C(C=O)C1(C)C.C1(CO)CC2(CC2)C1 69714,c1(OCC(=O)NC(CC=C)CNC(C2C3CC4C(C3=O)C24)=O)nc(O)nc(O)n1 69715,Cc1cccc2c1CC(C(=O)NCC=CCNC(=O)CC1(C)CCC1)O2 69716,c1(C(N2CC3CC(NC(CCC(=O)NC)=O)C3C2)=O)onc2c1CCCC2 69717,C(=O)(C(C(=O)N1CCOC(C(=O)NC23CC(C2)C3)C1)OC)OCC 69718,C(=O)(CC(C)CNCc1snc(C)c1N)OC 69719,C1(O)(CC(N2CCC(OCC(=O)NCC3ON=C(C)C3)C2)=O)CCCOC1 69720,Cc1cc(C(N2CCC(C)C2C(=O)NC(C)(C)CCCO)=O)[nH]c1C 69721,C1(OC)CN(C(c2cnn(C)n2)=O)CC1NC(=O)C(C)C 69722,c1(C(=O)NC2CCCN(C(c3nccc(C)c3)=O)C2C)cc2cc(Cl)ccc2[nH]1 69723,Cc1cc(C(=O)NCC=CCNC(C2CC3CC(=O)C2C3)=O)nc(C2CC2)n1 69724,C1(F)(C(=O)NCCCOCCCNC(c2c(C)ncnc2)=O)CCCCCC1 69725,C(=O)(CC(C)P(C)(C)=O)N1C(CNC(Cc2c(C)non2)=O)CC(O)C1 69726,c1(C(=O)NCC2CC(=O)NC2)cc(Cl)c(F)cc1[N+](=O)[O-] 69727,CC(C)(C)CC(O)C(=O)NC(CNC(c1cc(C(N)=O)[nH]n1)=O)CO 69728,N1(C(C2(OCC)CCOC2)=O)CCC(C2(NC(=O)Cn3ccc(C)n3)CC2)C1 69729,CN1CCCC(CCC(=O)NC2(C3CN(C(c4ccon4)=O)CCO3)CC2)C1 69730,C1(CCNC(C(COC)C)=O)CSCCN1C(=O)CC1(O)CCCC1 69731,C1(F)(C(N(CC(C)N(C(=O)CC2CCN(C)CC2)C)C)=O)CC=CCC1 69732,CC1(CC(N2CCC(OCCNC(=O)Cc3ccc(Cl)cn3)C2)=O)CCOCC1 69733,n1(CC(N2CCCCC(NC(C3(O)CC(C)(C)C3)=O)C2)=O)cnc2ccccc12 69734,C(=O)(C(CC(C)(C)C)NC(=O)CNC(C1CC1C)=O)N1CC(OC)C(O)C1 69735,c1(C(=O)NC2CC(C)CN(C(c3csc(C#N)c3)=O)C2)cnc2ccccn12 69736,C1(NC(CC(=C)C)=O)CC2CN(C(=O)C#CC(C)(C)C)CC2C1 69737,C1(CNC(COCCC(C)C)=O)CN(C)CCN1C(=O)C(C)Cn1ccnc1 69738,C1(NCC2(SC)CCC2)CC2CN(Cc3cccc(C#N)c3)CC2C1 69739,N1(C(C(=COCC)C#N)=O)CC2(C1)CN(C(c1cncc(F)c1)=O)CC2CO 69740,O=C(C(Cl)=CCl)NC1(C2CCCN2C(C2CC2c2ccncc2)=O)CC1 69741,C1(C(=O)NCCCc2cccs2)CCCN1C(=O)C(c1ccccc1)O 69742,C1(C(=O)NCC(C(=O)OC)OC)C2CCC(C2)N1C(C1C=CC=CC=C1)=O 69743,c1(C(N2C(CC(=O)Nc3ccc(N(C)C)nc3)CC2)=O)ncc(F)cc1N 69744,CC1(C)CN(C(=O)C(c2cccc(F)c2F)(F)F)CC(CNC(=O)C(C)(F)F)O1 69745,N1(C(c2c(C)cc[nH]2)=O)CCC2(CC1)CC2CNC(=O)C=Cc1ccc(Cl)cc1 69746,CCS(=O)(=O)CCN=c1[nH]c(N2CCOCC(CNC(C)=O)C2)nc2c1CSC2 69747,CC1COCC1(Nc1ccc(-c2nncn2C)cc1)NCc1ccccc1Cl 69748,C(CS(=O)(=O)CC(=O)NC1COCC1C(=O)NOCC1(C)CC1)OC 69749,C(=O)(C(C(C)O)N(C)C)NCC(C)CNC(=O)CCNC(c1ccsc1)=O 69750,C12(C(N(CC)Cc3cnnn3C)=O)CC(CN1C(=O)CC1CCC(=O)N1)C2 69751,C12(NC(c3ccc(F)c(O)c3)=O)CCC(C(N3CCC3CO)=O)(CC1)C2 69752,C(CC(C)(C)CNC(c1cc(C2CC2C)on1)=O)NC(c1cnc(SC)s1)=O 69753,c1(C(N(CC(CNC(COC(C)=O)=O)C)C)=O)ccc(N2N=CCC2=O)cc1 69754,C1(CC(=O)NCCCOC)C2CN(C(C3CCCOC3)=O)CC12 69755,C1(CN(CCCNC(Cc2cn(C(C)C)nc2)=O)C)CC2(CCC2)CO1 69756,C(c1ccc(=N)[nH]c1)=CC(=O)N(CC(C)NC(=O)COc1ccc(Cl)cc1)C 69757,Cn1cc(S(=O)(=O)N2CCN(C(=O)CSC3CC3)C3CC23)cn1 69758,C1(C(=O)NCc2ccc(C(N(CC(C)O)CC(F)F)=O)s2)CCCCCC1 69759,N1(C(C2(COC)CC2)=O)CC(NC(c2cnccn2)=O)C(SC)C1 69760,c1(SCC#C)cccc(C(N2CCC(CNC(c3cncc(F)c3)=O)C2)=O)c1 69761,N1(C(C)C(=O)NC2(CNC(=O)CCN3CCC(F)C3)CCC2)CCCC(O)C1 69762,C1(C)(C(=O)NCc2cccc(CNC(C(C)(C3CC3)OC)=O)c2)CCCNC1=O 69763,C1(C(N(CCCC(=O)N(C(CC)COC)C)C)=O)CC(=O)NC(=O)N1 69764,c1(CNC(C=C(C)C(C)C)=O)cccc(CNC(C2(C)CC3CC3C2)=O)c1 69765,CCCCCCC(O)CCC(=O)NCC1CC2CCC1N(C(=O)C(C)(C)CF)C2 69766,c1(C(=O)NC2C(NC(c3c(Cl)cccc3Cl)=O)COCC2)cnc2ccsc2c1 69767,c1(C(c2n(C(CC)C)nnn2)NCCC(=O)NC2CC2)cc(Br)c(C)nc1OC 69768,c1(NC(C2CC3(CCC3)C2)C)cnc2ccccc2n1 69769,c1(CC(N2CCC(CN(C(c3nnc(C)s3)=O)C)C2)=O)ccc2nn(C)cc2c1 69770,N1(CC)CCC(N=c2cccc(S(=O)(=O)NCCNC3(C)CCOC3)[nH]2)CC1 69771,N1(C(=O)C(Br)Br)CCCC(Cn2cc(CN3CCCC3C(=O)O)nn2)C1 69772,c1(C(C(=O)N(C(CC)C)C)N(CC(=O)NC)CC)ccn2nccc2c1 69773,c1(CC)noc(CCC(=O)NCC2CC(CNC(c3ccc(CO)o3)=O)CO2)n1 69774,C#CCC(CC#C)C(=O)NC1CC(CCNC(c2ccc(C)c(Br)c2F)=O)C1 69775,N1(C(C(C)c2ccsn2)=O)CCC(C2CC2)(CNC(C2CN(C)C2)=O)C1 69776,N1(CC)CC(C(N2CC(n3cc(-c4cccc(C(=O)O)n4)nn3)C2)=O)NC1=O 69777,C1(NC(=O)COCCNC(C2CS(=O)(=O)C2)=O)CCCC1C1CC1 69778,c1(CC(N2CC3C(CNC(c4occc4Cl)=O)(C3)C2)=O)ccc(O)c(Cl)c1 69779,N1(C(C(c2scc(C)n2)C)=O)CCC(NC(C23CCC(CC2)OC3)=O)CC1C 69780,Cc1ccc(CC(=O)NCC2CN(C(c3ccncn3)=O)CC(C)(C)O2)c(F)c1F 69781,CCC(CCOC)C(=O)N1CCN(C(c2cnncc2O)=O)CC1CCO 69782,N1(Cc2n(C)ccn2)CCC(F)(C(=O)Nc2nc(N(C)C)sc2)C1 69783,N1(C(CC2N(C)CCC2)=O)CCC(OCCNC(C2CCSC2)=O)CC1 69784,C1(C(F)F)(CNC(=O)C=C2CCCCC2)CCN(C(=O)CC2CC3CC3C2)C1 69785,c1(C(=O)NCC(C)NC(C2(CC=C)CCCCC2)=O)nc2nc(C)cc(C)n2n1 69786,CCC(C)(C)C(C)CC(=O)N1CCOC(CN(C)C(c2cc(C)nc(C)c2)=O)C1 69787,C(C(=O)NOCc1ncccc1C)(C1(C)CC1)NC(c1ccc(C)o1)=O 69788,c1(CNC(N2CCCCCC2C(F)(F)F)=O)ccc(Cl)c(F)c1 69789,C1(n2cc(C(C3CC=CCC3)=O)nn2)CCN(C(=O)C(F)(F)C(F)F)CC1O 69790,C(=O)(C1=CSCCO1)N(C1CN(C(c2csc(C(N)=O)n2)=O)CC1(C)C)C 69791,C(=O)(CCS(C)(=O)=O)NC1C=CC(CNC(C(C)O)=O)C1 69792,C(=O)(CCC(C)NC(=O)C(C)(C)CNC(C)=O)NC(CCC)C 69793,c1(C(N2C(C)CN(C(=O)CCOC3COC3)CC2)=O)ccc(S(N)(=O)=O)o1 69794,S(=O)(=O)(c1cc(C(=O)NCCN(C(c2ccc(N)cn2)=O)C2CC2)co1)NC 69795,C(CN=c1cc(NCC2(CN3CCOCC3)CCCCC2)nc[nH]1)(C(C)C)OC 69796,C#CCC(C)(CNC(c1cc(C)ncn1)c1nnnn1CCCCCC)CO 69797,c1(C(=O)NC2(CNC(CC3(OC)CC3)=O)CCCCCC2)ccc2nc(C)oc2c1 69798,c1(C2N(C(c3cc(Cl)ccn3)C(=O)NCCSC)CCC2)cc(F)cc(F)c1F 69799,C#CCC(C)(CC)C(=O)NCC(CNC(c1c(C)[nH]c(C)c1C)=O)OC 69800,Cc1cccn2cc(C(=O)NC3CCN(C(=O)C(F)CC4CC4)C3C)nc12 69801,c1(CC(=O)NCCC(C)N(C(C(C)SCC)=O)C)c(C)cc(OC)cc1C 69802,C1(NC(Cc2n(C)ccn2)=O)CCC2CN(CCCCc3ccccc3)CC2C1 69803,c1(C(=O)NCCCCNC(c2nccc(C(N)=O)c2)=O)ccc2n[nH]cc2n1 69804,CCC(C(=O)NC1(CF)CN(C(C2CCSC2)=O)C1)C(C)(C)CC 69805,c1(CNCCC(C)OC)ccc2nc(C)n(C)c2c1 69806,c1(OC)ccc(NC(=O)C(=O)NCc2ccsn2)cc1OC 69807,C(C(=O)NC1CCC(NC(C2CCCCN2C(N)=O)=O)CC1)(C(C)C)OCC 69808,Cc1cnccc1N1CCN(c2nnc(C3CC3)n2CCc2ncn(C)n2)CC1 69809,N1(C(c2cc(CC)[nH]n2)=O)CC(NC(c2cc(C)nc(O)c2)=O)CC12CCCC2 69810,CCC(Cc1ccccc1)CC(=O)NC1CC(CNC(=O)CCCc2nccs2)C1 69811,CC1=NOC(C(=O)N(CCC(C)NC(c2snnc2C(C)C)=O)C)C1 69812,CCCCC(CNC(C1CCN(CC)C1)=O)NC(=O)C(C)(O)c1ccccc1 69813,C1(NC(Cc2c(C)nn(C)c2)=O)C2CCC(C2)C1C(=O)NC1CN(C(N)=O)C1 69814,C1(C(=O)NC(C=CC(=O)NC(C)Cc2ccncc2)C)CCC(C)(C)O1 69815,C=CC(C)(O)CC(=O)N1CCOCC1CNC(=O)CC(C)c1ccncc1 69816,C1(C(C)NC(=O)C=C2CCCCC2)CCCN(C(=O)Cc2ccc(Cl)cn2)C1 69817,C1(OC)CC(C(N(C(C(C)NC(C2CC(SC)C2)=O)CO)C)=O)N(CC2CC2)C1 69818,CC1CC(NC(C2C(C)OCCN2C(=O)CC2(C)CCCCC2)=O)C(C)CN1C 69819,C1(NC(Cn2c(C)ncc2)=O)CCCN(C(c2cncc(C3CC3)c2)=O)CCC1 69820,C1(C(C(N2CC(CO)(NC(C3(CO)CC3(F)F)=O)C2)=O)O)CCCCCC1 69821,CN1CCN(CCC(N2CC3C(NC(=O)COc4ccc(Cl)cc4)C3C2)=O)CC1 69822,C1(C(N2CCC(N(C(=O)CS(=O)(=O)NC(C)(C)C)C)C2)=O)CC(=O)NC(=O)C1 69823,CC1(C)CCCN(C(=O)C(F)C(F)(F)F)C1C(=O)NCC1(O)CC(O)C1 69824,c1(NC(=O)NCC(C2CCCCCC2)C)ccc2c(c1)N(C)CCO2 69825,N1(C(=O)NCCc2cccc(C)n2)C2CCCC1CC(O)C2.c12ccccc1C2 69826,O=S(=O)(c1cnn2ccc(N3CC4CCC4C3)nc12)NCc1sncc1Br 69827,C(CCCC(=O)NC1(C(=O)NC2CC3C=CC2C3)CCC1)OC 69828,O=S(=O)(c1cncc(Br)c1)NCC1CC2CC2N1CC12CCCN1CCC2 69829,C(=O)(CCC(C)=O)NC1C(CCC)C1.C1(C)CCN1 69830,Cn1cc([N+](=O)[O-])c(-c2nnc(-c3ccn(C)n3)o2)n1 69831,c1(CC(=O)NCCNC(c2nn(CC)c(C(F)(F)F)c2)=O)ccc(C)c(F)c1F 69832,N1(C(=O)Nc2ccccn2)CCC2(CCN(S(=O)(=O)c3cncc(Br)c3)C2)C1 69833,c1(NC(c2n(COC)ncc2)=O)ccc(Br)c(OC(F)(F)F)c1 69834,C(=O)(C(=O)N=c1ccn(C2CCOC2)[nH]1)NCCC1CCC(C)O1 69835,N1(C(C2C(C)C2C)=O)CC2CCC1CN2C(=O)CC1CN(C(C)(C)C)CC1C 69836,Cc1ccc2cc(C(=O)NCc3cccc(-c4ccccc4)n3)[nH]c2n1 69837,C(=O)(CCCCCF)N(C(C(=O)NC1CCCN(CC)C1)C)C 69838,n1(CCC)nnnc1C(C)(CC1CCC1)NCc1nc(C)co1 69839,CC1C=C(C(=O)NCC(c2ccccc2)NC(=O)C=Cc2ccc(F)cc2)CC1 69840,N1(C(CC(C)OC)=O)CCCC12CCN(C(C1CCN(C)CC1)=O)C2 69841,c1(C(N(C2CCCC(NC(=O)C(C)(F)c3ccon3)C2)C)=O)[nH]ncc1C#N 69842,c1(C(=O)NCC(C)N(C(C2CCC(C)(CC)O2)=O)C)cnn2c1NCC(C)C2 69843,C1(C(=O)OC)CCN(C(=O)CC2(C)CCN2C(=O)COCC2CCC2)C1C 69844,n1(CCC(N2CC(CC)C(NC(=O)COC)CC2)=O)ncc2cc(Br)ccc12 69845,Cc1cc(NC(=O)CC2CCN(C(c3cn[nH]c3)=O)C2)cc(C#N)c1 69846,C(=O)(CCCC(C)(C)C)N(CC(C)(C)CNC(=O)CCCOC(=O)CC(C)C)CC 69847,N1(C(C2N(C(CN(CCOC)C)=O)CCOCC2)=O)CCCN(C)CC1C 69848,c1(C(=O)NC(C(C(C)C)Nc2nnccc2C#N)C)c(Cl)cccc1Cl 69849,C1(CCC(=O)CCSc2cscn2)CCNCC1.CC(=O)O 69850,Cc1n[nH]c(C)c1CCC(=O)NC(C)CNC(=O)CC1CC1C(F)(F)F 69851,C(CC(C(C)(C)C)NC(C1(O)CC1)=O)N(C)C(c1cnc(Cl)cc1N)=O 69852,c12ccc(cc1OC)C(=O)OCCS2.c1(C2C(C(=O)OC)C2)ccco1 69853,N1(C(C2(C)CC(NC(=O)C(O)Cn3cncn3)C2)=O)CC2(C1)NC(=O)NC2=O 69854,C1(CNC(C(CC2CN(C(CP(C)(C)=O)=O)C2)F)=O)CCC2(CCC2)O1 69855,Cc1ncc2n1CCC(C(=O)NC1COC3(C1)CN(C(C14CC(CO1)C4)=O)C3)C2 69856,CCC(C(=O)NCC1CC(O)CN1C(=O)C1=CCC1)C(C)(C)CC 69857,c1(C(N2CCC3(CCCC3)C2)C(=O)NCC(F)F)ccc2c(n1)CCC2 69858,N1(C(COC(CC)C)=O)C2CCC1CC(C(=O)Nc1cc(C)nc(C)n1)C2 69859,C=CCCC(C(=O)NCC(C)CCC)NC(=O)C(C)NC(=O)OC 69860,C1(N(CC(=O)N(C)Cc2cn[nH]c2)C(c2ccoc2C(=O)O)=O)CC(O)C1(C)C 69861,C(=O)(CS(F)(F)(F)(F)F)NCC(C)NC(c1ncsc1C(F)(F)F)=O 69862,CC1(C2CC2)CCN(C(=O)C(Cc2cc[nH]n2)NC(=O)COC2CCOCC2)C1 69863,N1(CC(=O)N(C2CCC(CNC(=O)CC3COCC3O)CC2)C)CCCNC1=O 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69882,C(C)(CCC(C)C)(c1nnnn1CCN1CCOCC1)NCc1nc(C)c(C)s1 69883,Cc1nn(CC(=O)NCC(C)(F)CNC(=O)C(C)(C)CC2CC2)c(=O)o1 69884,CC1(C)C(NC(C2CC3CC(=O)C2C3)=O)C2CCCN(C(=O)CCC3CCC3)C12 69885,N1(C(CC)=O)CCC(COCCNC(=O)C(=O)Nc2nnc(C)o2)C1 69886,C1(NC(CSCC#C)=O)CC(CNC(c2cc(C)n(C)c2C)=O)C12CCC2 69887,c1(C(=O)NC2(CCNC(C(C(CC)O)C)=O)CC2)cc2oc(Br)cc2s1 69888,C#CCCN=C(NCCc1ccc(C)c(O)c1)NC1CCS(=O)(=O)C1 69889,N1(C(C2(C)CC(C)C2)=O)CCC(CCCCNC(C2(C(F)(F)F)CCC2)=O)CC1 69890,c1(C(N2CC(NC(CC3(C=C)CCCCC3)=O)C(C)C2)=O)cccc2nccn12 69891,CC1CN(C(C2(c3ccno3)CC2)=O)CCCN1C(=O)CC(C)(C)C#N 69892,CC1=NC(C)(CNC(C2(CNC(C3CCNC3=O)=O)CCCO2)=O)CS1 69893,c1(OC)ccc(C(=O)NC(C2CN(C(c3sccc3F)=O)C2)C)c(OC)n1 69894,C1(N(C(c2cc(C)n(C)n2)=O)C)CN(C(=O)Cc2c(O)ncnc2O)CC1(C)C 69895,C1(N(C(c2c(SC)cn(C)n2)=O)C)CCN(C(=O)C(C)(C)c2cscn2)CC1C 69896,C12(C(=O)NCCC(C)N(C)C(c3cccs3)=O)CCCC(CCC1)C2=O 69897,c1(NC(C2N(C(CC(C)SC)=O)CCCC2)C)cc(O)nc(O)n1 69898,C1(C(=O)NCC(n2cc(-c3ncoc3C3CC3)nn2)C)CCC(F)C1 69899,c1(OCC)ccccc1-c1nc(C2COCCO2)n(C2CCOC2)n1 69900,C1(NC(C(COC)C)=O)(CO)CCCN(C(c2ccn(CC(F)F)n2)=O)C1 69901,c1(SCC)cc(Cl)ccc1C(=O)NCC1CC(O)(CNC(C2CCS2(=O)=O)=O)C1 69902,c1(C(N(C2CCN(CCc3ccccn3)CC2)C)=O)cc2ccsc2[nH]1 69903,c1(CN2CC(NC(c3scc(C)c3)=O)C(O)C2)cccc(S(C)(=O)=O)n1 69904,N1(C(c2ccc(N(C(C)=O)C)cc2)=O)CCCC(CO)(NC(=O)CS(C)(=O)=O)C1 69905,N1(C(c2c(CC)oc(C)c2)=O)CC2CN(C(c3cccc(O)n3)=O)CC(C1)O2 69906,C1(N(C(CC(=O)N(C)C)=O)C)CCCCN(C(C2C3CCOCC23)=O)C1 69907,C1(CC=C)(NC(=O)COC(C)=O)CCN(C(c2cc(O)nn2C)=O)C1 69908,n1(CCN(C(=O)C(CC2CCOC2)OC)CC)cc(C(O)C2CC2)nn1 69909,C#CCC(CC(F)F)C(=O)NCC(F)(C(=O)N(C(C)CN(C)C)C)C(C)C 69910,Cc1cc(NC2CCCN(C(c3ccnc4c3ncn4C)=O)C2)ncc1[N+](=O)[O-] 69911,n1(CC(=O)OC)cc(C(N(C(c2ccc(Br)o2)=O)CC)C2CC2)nn1.C1CCOC1 69912,C(C(C)C)(C(O)C(=O)NC1CCC(N(C(=O)Cn2cncn2)C)CC1)OC 69913,c1(CCC(N2CC(CC(C)NC(C3CC(F)CN3C)=O)C2)=O)ccc(Cl)nc1 69914,CC(CC(=O)NCC=CCN(C(=O)NC(C)(C)C)C)OCCOC1CC1C 69915,c1(OC(CC)C)cccc(=NC(=O)Cc2cccc(CN=S(C)(=O)N(C)C)c2)[nH]1 69916,N1(C(c2ccc(NC)cc2)=O)CC(C(=O)Nc2ccsc2CO)CC(C)C1 69917,Cn1nnc2c(N3CC=CC(NC(=O)Cn4ncc5cccnc45)C3)ncnc12 69918,C(C(CC(C)C)C(=O)NCCC1CC1)NC(c1c(C)noc1C)=O 69919,Cc1n[nH]c(C)c1CC(N1CCC(OC2CN(C(c3cnc(S)[nH]3)=O)C2)CC1)=O 69920,C1(NC(C2(SC)CC2)=O)CN(C(C2C3CCCC23)=O)C(C)(C)C1 69921,c1(C(C(=O)NC(COC)CNC(=O)CCOCC(F)F)O)ccc(F)c(Cl)c1 69922,N1(C(CCN(CCC)C)=O)CCN(C(C2C=CC=CC=C2)=O)CC1C 69923,C=CCCCC(C1CC1)NC(=O)C=CC(=O)OC.C1(=O)C(C)C(C)N1CC 69924,c1(C(=O)NC2CCN(C(C(CCC)C)=O)CC2)sc2ccccc2c1Cl 69925,C1(NC(C(CC(=C)C)C)=O)CN(C(c2cc(C3CC3)nn2C)=O)CC2CCCC12 69926,c1(OC)ccc(C(CNC(c2cncc(CO)c2)=O)NC2CC(CN)C2)cc1 69927,N1(C(C(=O)NCCCN(C(CC)C)C)=O)CCC(F)(C#N)C1 69928,N1(C(c2c(C)c(Br)cnc2)C(=O)NCC(C)C)CC(C#N)C2(CCC2)C1 69929,c1(C(N2CC(CCNC(c3ccc(OC)c(O)c3)=O)C2)=O)c(F)ccc(F)c1Cl 69930,C(=O)(CCS(=O)(=O)C(F)(F)F)N(CC(C)O)CCNC(C1CCCCO1)=O 69931,c1(OC(C(=O)NCC(CC)NC(C2CC(O)C2)=O)C)ccc(Br)cc1 69932,c1(C(=O)NCC(CC)NC(c2coc(C3CCCC3)n2)=O)ccn2ncnc2c1 69933,c1(C(=O)NCCCCCCNC(CCCC)=O)c(Cl)ccc2ccoc12 69934,c1(C(N2CCC(NC(c3cc(C)sc3)=O)CC(O)C2)=O)ccc2oc(N)nc2c1 69935,c1(C(=O)NC2CCCN(C(COc3ccc(N)cc3)=O)C2)cccc([N+](=O)[O-])c1 69936,c1(NCC2CC(NC(C(C=CCCC)O)=O)C2)ccc([N+](=O)[O-])cc1S(C)(=O)=O 69937,C1(NC(c2c(C)nn(C(C)C)c2)=O)CC2(C1)CN(C(=O)C(C)C(C)C)C2 69938,C12(NC(=O)C(CC3CC3)NC(C3CC4CC3CC4=O)=O)CCC(C1)C(O)C2O 69939,N1(C(C(C#C)(C)C)=O)CCC(NC(C2CC2=C)=O)C(C)(C)C1 69940,S(=O)(=O)(c1cccc(=NCCCOCCO)[nH]1)NCCN1CCC(=O)NC1=O 69941,C1(NC(c2c(NCC)scn2)=O)CCCCC1CNC(=O)C(C)(C)C 69942,C1(C(=O)NC2CC(N(C)CC)C2)CN(C(=O)Cc2cc(C)nn2C)CC12CC2 69943,C1(C(CN)NC(C2(CF)CC2)=O)CCCCC1.CCCC(C)N(CCC(=O)C1CC1)C 69944,c1(C(=O)NC2CC(C)CN(C(=O)CC3CCCC3)C2)c(F)cc(F)cc1Br 69945,CCCC(C)(CC)C(=O)NCC1CCCCC1NC(C1CCCC1S(C)(=O)=O)=O 69946,c1(OC)cc(C(N2CCN(C(=O)COCC3CCCC3)C(CF)C2)=O)cc(F)c1 69947,C1(CC(=O)N(CCCNC(=O)C(C)NC(N)=O)CC)COCCOC1 69948,CC1=C(C(=O)NC2CN(c3ccccn3)C2)CCO1.C12CC1C(=O)N2 69949,C1(N(C(C2COC(C)C2)=O)CC)CCCN(C(=O)Cc2csc(Cl)c2)CC1 69950,C12(C(=O)NCC3(F)CN(C(CS(=O)(=O)NCC)=O)C3)CCCCC1NC(=O)CC2 69951,CCC(CC)(CC)C(=O)NCCC1CC(NC(c2ccc(C#N)c(Cl)c2)=O)C1 69952,Cc1cc2[nH]c(=O)c(C(=O)NC(C)CN(C)C(C3CCCC(C)CC3)=O)cn2n1 69953,C1(CC(F)(F)F)C(C(=O)OC)CCCN1C(=O)NCCNC(N)=O 69954,CC(C(=O)NC1(C(=O)NC(c2ccc(F)cn2)C)CCN(C)C1)C(F)F 69955,N1(C(c2ccc(CNC(C)=O)o2)=O)CCC2CN(C(=O)Cc3cncn3C)CC12 69956,c1(C(CC)C)ccc(C(=O)NCC2(C)CCCN2C(c2cnn(C)n2)=O)c(O)n1 69957,c1(OC)cccc2c1CCN2c1nnnn1C.C12C3CN(CC13)c1ccnc(n1)N2 69958,N1(C(C(C)OCC(C)C)=O)CC(NC(=O)CCNC(c2ccoc2)=O)CC(O)C1 69959,Cc1nc(C(=O)NCC2CC2NC(=O)CCC=CBr)cn1C(F)F 69960,C=C=CCCC(=O)NC1CCC(C)(CNC(=O)CCN(CCCCC)C(C)C)C1 69961,C#CCC(O)C(=O)N(C1C=CCN(C(=O)CC(F)(F)F)C1)Cc1ccccc1 69962,c1(CNc2c(C(=O)NC3CCOCC3)n[nH]c2)c[nH]c2cc(Br)ccc12 69963,c12cccc(c1)C(=O)NC2.CC1(CN2CCSCC2)CCCC1 69964,N1(C(C(C)=CC(C)(C)C)=O)CC(=O)NCC1C(=O)NCCCCCF 69965,CC(N=c1[nH]nc(C2CCCC2)s1)C1CCN(C(=O)Cc2ncn3c2CCC3)C1 69966,C(CC(C)(C)C)(C(=O)NCC1CCC1)NC(C(CCCC)O)=O 69967,c1(CNC(C2CNC(=O)N2)=O)ccc2c(c1)CCC2NC(=O)C=Cc1cn[nH]c1 69968,C(=O)(C1CCCc2cccnc21)NC1CCCN(C(c2ccc(C)o2)=O)CC1 69969,C(=O)(CS(=O)(=O)CCO)NC(C)CCCNC(C1CCCOC1C)=O 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70005,Cc1ccc(CC(N2CC(NC(C3(F)CC=CCC3)=O)C(C(F)(F)F)C2)=O)cc1 70006,c1(-n2c(=O)ccc(C=CC(F)(F)F)c2)cn(C2c3ccccc3CC2CCO)nn1 70007,c1(C(N2CC3(C(C(=O)Nc4ccc(C)c(I)c4)C3)C2)=O)cnn2cccc(F)c12 70008,c1(OC)nc(C)ncc1C(=O)NC(C)(C)CN(C(=O)C(C)CC1CCCO1)C 70009,C12CCC(N(C)C)(CC1)C2=O.c1(C(=O)OC)ccc(C2CCC(=O)N2)cc1 70010,Cn1cc2c(C(N3CC4CCCN(C(=O)Cc5cc[nH]n5)C4C3)=O)cccc2n1 70011,C(C(N=c1ccc2nnnn2[nH]1)C(C)C(C)C)NC(c1c(C)nc(CO)nc1)=O 70012,C1(NC(C(C2CC2)SC)=O)CCCCCC1NC(=O)CC#N 70013,N1(C(c2c(C)nc(CCC)s2)=O)CCC(NC(C2CCCCN2CC)=O)C(F)C1 70014,O(NC(=O)CN(C(=O)CCOCC(C)C)CCC)CC#C 70015,CCCCCCC(F)C(=O)NC(C)CNC(=O)CCOc1ccccc1C 70016,C#CCC(CC(=O)NC(C)C(=O)NC)NC(C1CN(C)C1)=O 70017,O=C(C(CCC1CC1)c1ccccc1)NCCC1CCN1 70018,c1(C(N2CC(N(C(CCCCN(C)C)=O)C)C(F)C2)=O)ccc(F)c(N)c1 70019,Cc1ccc(CNC2(Cc3ccc(Br)cc3)CC2)c(O)n1 70020,c1(C(N2C(C(=O)Nc3cc(Cl)ccc3CO)C=CC2)=O)cc(Br)cc2[nH]ncc12 70021,CCCC(CC)CCC(=O)NC12CC1CN(C(c1nnc(O)nc1O)=O)C2 70022,c1(C(N2CCCC2C2(C)CC2)C(=O)NCC(=C)C)cnn(-c2nccs2)c1 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70040,c1(C(=O)NCC2C(NC(=O)CCc3ccncc3)CC2)n[nH]c2c1COC2 70041,c1(C(=O)NCC2CCC(NC(=O)C(Cl)=CCl)C2)cn2ncccc2n1 70042,N1(C(C(C(COC)C)C)=O)CCN(C(=O)Cc2cc[nH]c2)C2(CC2)C1 70043,c1(C(=O)NC2(CC=C)CCN(C(C3CC3C(F)(F)F)=O)C2)ccc(Cl)c(C)c1 70044,C(c1nc2ccccc2o1)=CC(=O)NC(C)CNC(c1ccc2ocnc2n1)=O 70045,C(CC(C(=O)N(C1CCCC1)C)NC(c1csnn1)=O)=CC 70046,C1(CN(C(c2cnc(C(C)O)s2)C(=O)NC2(C)CC2)CC=C)CCCOC1 70047,CC(C)C(CC(=O)NCCCc1cc[nH]n1)NC(=O)C(c1ccn(C)n1)C 70048,CCC(C)(C)C(O)C(=O)NC1(C2CCN(C(C3CCCN3C=O)=O)C2)CC1 70049,Cc1cc(C)c(C(=O)NC2CN(C(=O)CC3(CO)CCCC3)CCC2C)c(C)n1 70050,C1(NC(c2csc(O)n2)=O)CC2CC1N(C(C1CN(CC(F)(F)F)C1)=O)C2 70051,c1(Cn2cc(N(CC(CC)NC(=O)C3CC3)CCOC)nn2)cccc(F)c1 70052,C=CCC(CC=C)C(=O)N1C2CCC1C(CNC(=O)C(C)(C#N)CC)C2 70053,CCC(C(=O)NC(C)CCC(=O)NCCN(C1CCC1)CC)C(F)(F)F 70054,C1(C(=O)NCC(=O)NCCN(C(=O)CC(F)F)CC(C)O)CCOCC1 70055,CC(C(=O)NC(CC1CCC1)C(=O)NCCc1cnco1)C(F)(F)F 70056,c1(CC)ccnc(C(=O)NC2COCC2N2CCN(C(C3CC3C#N)=O)CC2)c1 70057,N1(C2c3c(c(C)ccc3)NC2=O)CCC2(C=Cc3ccccc3O2)C1.CCOC 70058,C1(C(=O)NC(C(C2CC2)OC)C)CC(OC)CN1C(=O)OC(C)(C)C 70059,N1(CC)CCC2(CCC(O)C2)C1.c1(C(=O)OCC)c(N)c(C#N)cn1CCl 70060,N(C1CCOc2ccccc21)(C(=O)CC1CC1C1CC1)CCCF 70061,n1(CCNC(C2(c3ccncc3)CC2)=O)cc(CCCCCC2CC2)nn1 70062,N(C(=NCCC(C)(C)C)N(C)Cc1noc2ccccc12)C(C=C)C 70063,c1(C(=O)NCC2CCCCN2C(=O)CCC2CC2CC2CC2)nnn2c1CCC2 70064,C(=O)(CC(C(F)(F)F)P(C)(C)=O)N1CCC(N(C(=O)C#CC2CC2)C)C1 70065,n1(COC)nc(Br)cc1C(c1nnnn1C)NC(CC(N)=O)C1CC1 70066,CCC(CCCC(=O)NCC1Cc2nccn2C1)NC(=O)Cn1cccnc1=O 70067,c1(COC)csc(C(=O)NCCN(C(=O)C(=O)N(C)C)CC2CCCC2)c1 70068,CCCC(CC)C(=O)NC1CCC(NC(=O)COCC=Cc2ccccc2)CC1 70069,c1(C(=O)NCCCN(C(C(n2ccc(C)n2)C)=O)C2CC2)cccc(C)c1C 70070,N1(CC)CCOCC1C(=O)NC(C(=O)N(C)CCC1CN(C)C1)C1(O)CCC1 70071,C(=O)(C(O)CC(N)=O)NC1C(C)CN(C(=O)CCCN(C)C)C1 70072,N1(C(C(CC=C)(C)C)=O)CCC2(CC1)CC(CNC(C1CC(C)CC(C)C1)=O)C2 70073,CCS(=O)(=O)c1cnc(O)c(C(=O)NC2C3CN(C(=O)CC4CC=CC4)CC23)c1 70074,C(=O)(C#CCC(C)C)NCCN(C(=O)CCCCN(C)C)CCC 70075,C(C(=O)NCC1C(OCC(=O)NC2(CO)CCCC2)CCCC1)(C(C)C)OCC 70076,CC1CCN(C(C2CCS(=O)(=O)N2)=O)C(CNC(C2CC(=O)C2C(C)(C)C)=O)C1 70077,N1(C(C(CCCC)F)=O)CCC2CN(C(C3CC3C(F)(F)F)=O)CC2CC1 70078,Cn1nccc1CCNC(=O)CCC1(NC(C2CC2c2ccoc2)=O)CCCC1 70079,C(C)(C)(CC(F)C(=O)NC1CCCOC1)NC(C(C)SCC)=O 70080,c1(OC)ccccc1C(C)CC(=O)N(C1CC(NC(=O)Cc2c[nH]nc2C)C1)C 70081,c1(C(=O)NC2CC(NC(C3C(C)C3C)=O)C2)cccc2c1nnn2C 70082,CC1CN(C(C23CC(C2)C3)=O)CCC1NC(=O)CCc1nc(O)n[nH]1 70083,c1(C(=O)NCC2CCCCN(C(C(CC)F)=O)C2)ccc(S(N)(=O)=O)o1 70084,Cc1cc(=NC(C)CCNC(=O)C#CC2(C)CCCO2)[nH]c(C)c1C#N 70085,CCCCCC(C)NC(c1ccccc1Cc1ccccn1)=O 70086,N1(C(C(C(CC)O)C)=O)CCCC2(C1)CN(C(=O)CCc1ccccn1)CCO2 70087,c1(C(N2CCCC(C)(CNC(C(C)OCC=C)=O)C2)=O)coc(S(=O)(=O)NC)c1 70088,c1(NC(C(C)NC(c2cn(CC)nc2)=O)C(C)C)cc2nn[nH]c2cc1[N+](=O)[O-] 70089,C(=O)(C(C)(O)CC(F)F)NCCCOCCNC(c1ccc(NC(C)=O)o1)=O 70090,c1(CCNCC(COCC(C)C)O)coc(-c2ccccc2)n1 70091,O=C1Cc2cccc(C(=O)NC3CN(Cc4c(F)cc(I)cc4F)CC3O)c2N1 70092,C(=O)(N(CCC(=O)NC1CN(C)CCN1C)OC)N(C1CCCCC1CO)C 70093,N1(C(C2(OCC)CCC2)=O)C2CCC1C(CNC(=O)Cc1cccnc1Cl)C2 70094,N1(C(C(COC)O)=O)CCC(CC(=O)O)(NC(=O)OC(C)(C)C)C1 70095,c1(C(=O)NCC(C2CCCC2)NC(c2csnn2)=O)cccc2c1OCCO2 70096,c1(-c2scc(C)n2)ncc2cc(C)ccn12 70097,c1(C(N2C(CN(C)C(C3CCCOCC3)=O)COCC2)=O)cnn2ccncc12 70098,CCC(C(=O)NCCOCCN(C(=O)CC1CCC(O)C1)C)C(C)C 70099,c1(C(=O)NCC2(C(N(CC=C)CC3CC3)=O)CCC2)cnn(C=C)c1N 70100,C(=O)(C1=C(Cl)CCCC1)N(C1CCCN(C(c2cc(Cl)cn2C)=O)CC1)C 70101,C1(O)(CCNC(c2cc(C(C)=O)sc2)=O)CCN(C(=O)C(C)(C)C(F)F)CC1 70102,N1(C(COCC(=O)OC(C)(C)C)=O)CC2CC(C1)N(C(=O)CC1CC13CC3)C2 70103,N1(C(c2c(C(C)NC(c3ccsc3Cl)=O)noc2)=O)CCc2ccc(F)cc21 70104,C(CC(C)C(=O)N1CCC(C)(CNC(c2nn(C)cc2N)=O)C1)=CC 70105,N#Cc1cccc(NC(=O)C(CCC2CC2)NC(c2ccsc2Cl)=O)n1 70106,C(=O)(C(C)CC(C)(F)F)NCCCCCN(C(C1CC=C(C)CC1)=O)C 70107,C1(CCC(=O)OC)CNc2ccccc2C1Cn1c(=O)oc2ccccc12 70108,Cc1ccc(C(=O)NCC2C=CC(NC(C3CC(CC4CC4)C3)=O)C2)o1 70109,c1(CC(=O)N(CCN(C(=O)CCN2CCC(F)C2)C)C)ccccc1F 70110,C(=O)(C=CS(=O)(=O)CC)N1CC(CCn2cc(CC=C)nn2)C1 70111,c1(C(N(CCC(C(=O)NC(CC(=O)OC)(C)C)O)C)=O)cc(C)nc(O)c1 70112,c1(SCC#C)cccc(C(=O)NC(CNC(=O)C(c2cccs2)SC)CO)c1 70113,c1(OC)nc(C2=CCNCC2)ccc1C(N1Cc2cccc(O)c2C1)=O 70114,N1(C(=O)NC2(C(=O)O)C(C)C2)CCN2CCN(C(C3CCC(=O)N3C)=O)CC2C1 70115,C1(CNC(CS(C(C)C)(=O)=O)=O)CCC2CN(C(C3CC4CC4C3)=O)CCC2C1 70116,N1(C(C)C)CC2CN(CC34CCCC3C4)CCC12 70117,C1(NC(c2c(CC)nco2)=O)CCN(C(c2c[nH]nc2-c2cccs2)=O)CC1F 70118,c1(-c2nc(CCC)sc2)nc(C2OCCc3ccccc32)nn1CCCCO 70119,C1(CC(N2CC(COC)C2)=O)CC(C)(C)CN1C(=O)Cc1ccc(F)cc1 70120,c1(C(N2CCC(C)C(NC(c3ccoc3C3CC3)=O)C2)=O)cc(C#N)ccc1F 70121,Cc1nnc(O)c(C(=O)NCC(C)N(C(=O)C(C)Cn2cccn2)C)c1C 70122,N1(C(C(N2CCCC(C)C2)=O)=O)CCC(NC(=O)C(F)(F)c2cscn2)C1(C)C 70123,N1(C(C2CC3CC3C2)C(=O)NC(CC)C)CCC(C2CCCC2(C)C)C1 70124,c1(CC)cc(Br)c(F)cc1NC(=O)NCc1cn(-c2cc(F)cc(Br)c2F)nn1 70125,c1(CC)cc(=NC(=O)C2CC(NC(=O)CC3CCCCC3O)C2)[nH]n1C 70126,C1(C(=O)NCCCN(C(=O)C#CC2(C(F)(F)F)CC2)C(C)C)Cc2nncn2C1 70127,C12(C(=O)NC3(C4N(C(CC5(OC)CC5)=O)CCC4)CC3)CCN(CC1)C2 70128,c1(CN2C(C(N3CCC(C(N)=O)CC3)=O)CC2)c[nH]c2cccc(F)c12 70129,c1(C(N2CCC(NC(C(C)SC)=O)C(C)C2)=O)cccc2c1NCC2 70130,C(=O)(C(C(C)CC1CCOCC1)N(C)CC1CCCN(C)C1)NC(C)C 70131,C(C(=O)N(C)CC1CCOC1)(C1CN(C(=O)C(SC)SC)C1)OCC 70132,Cc1nnccc1C(N1CCC(CNC(=O)CN2CCCNC2=O)C1)=O 70133,N1(C(c2nc(C)[nH]n2)=O)CC(NC(=O)CCC(C)=O)CC1C 70134,C1(C(=O)NC(C)CCNC(=O)C(O)C2CCCC2)CCC(N=[N+]=[N-])CC1 70135,N1(C(C2=C(C)CC2)=O)CC2(C(N3CCOC(CCO)C3)=O)CC1CO2 70136,C1(C(=O)NC2CC(NC(C3N(CC)CCCC3)=O)C2)CC2(C1)CC(F)C2 70137,C1(CCC)CN(C(=O)C(=O)NCC2CC2)CCN1C(=O)COc1cccc(F)n1 70138,C1(N(CCO)C(=O)N)C2CN(C(=O)C(F)CC3CCOC3)CC12.Cc1cc(CO)on1 70139,C1(CNC(c2cc(OC)n[nH]2)=O)CN(C(C2CCN(C(C)C)CC2)=O)CCN1C 70140,CC1CCN(C(=O)OCC(C)(C)C)CC1.C1(C)(C)CS1 70141,C1(CC(=O)NCCCOCCNC(C(C(C)C)OCC)=O)CCCC2(CCC2)O1 70142,C1(C(=O)OC)CCC(NC(=O)CC2(C)CN(Cc3ccsc3SC)C2)C1 70143,C1(C(=O)NC(CC)CO)C(CNC(c2ccoc2Cl)=O)C1(C)C 70144,c1(C(=O)NC2CC(C)(NC(CC(C)CF)=O)C2)nc[nH]c2ncnc1-2 70145,c1(CC(C)N(C(c2ccc(C(Cl)Cl)cc2)C(=O)NC)C)c(C)nn(C)c1C 70146,CC(N=c1[nH]c2c(c(=NC3CCN(c4ccccc4)C3)[nH]1)CCC2)c1ccco1 70147,C1(NC(C2C(CC)C2)=O)CN(C(c2csnc2C)=O)CCC1C(F)(F)F 70148,c1(CC(N)C(=O)N2CCOCC2)ccccc1C1CC1 70149,C=CC(C)(O)C(=O)NCCCN(C)C(C1(c2cccs2)CC1)=O 70150,C1(NC(c2cccc(C3CCC3)c2)=O)C2CCN(C(C3CC=CCC3)=O)C12 70151,N1(C(C(C)OC)=O)CCN(C(c2ccc(-c3ccc(Cl)c(F)c3)o2)=O)C(CF)C1 70152,Cc1cc(C(=O)NCCn2c(C)ccc2C)c(Br)nc1C 70153,Cc1cc(C)c(C(=O)NCc2cc(C(=O)Nc3csc(C)c3)n[nH]2)s1 70154,c1(C(=O)NC2C(NC(c3c(OC)c(F)ncc3)=O)CC2)c(C)ccc(C)c1C 70155,c1(C(N2CC(C(=O)OC)C(O)CC2)=O)cccc2sccc12.C12CN(C(=O)O1)C2 70156,C1(NC(CN(C)CC)=O)CC2CC(NC(=O)CSc3n[nH]c(=N)s3)C2C1 70157,C(=O)(CC(F)(F)F)NCC(=O)NCCNC(Cn1c(C)ccn1)=O 70158,C1(C(=O)NCCCCCN(C(=O)C(C)(C)C(N)=O)C)CNc2ccnn2C1 70159,C1(C(=O)NCCN(C(=O)C(=O)Nc2ccccc2)CC)COCCN1C 70160,CCCC(CC(=O)NCCN1CCCCC1)NC(C1CC(CF)C1)=O 70161,C(CC(N)=O)(C(=O)N1CCCC(C(C)C)CC1)NC(CSCCC(C)C)=O 70162,C1(C)(C(N(CCC)C2CC2)=O)CC12CCN(C(C)Cc1cccc(Br)c1)CC2 70163,C1(C(=O)Nc2cc(CCC)[nH]n2)CC2(CCC2)CN1C(=O)Cc1ncccc1F 70164,N1(C(CC2CCC(=O)NC2)=O)CCC2(C1)CN(C(=O)COCC(F)F)CCO2 70165,CCCCCCC(C)(CC)C(=O)NC1CCC(NC(=O)CCc2nncs2)C1 70166,c1(C(=O)NC2(CNC(c3c[nH]c(=O)cn3)=O)CCOC2)cc(Cl)c(Br)[nH]1 70167,N1(C(C(=O)NC(CC)C)CC2C=CCC2)Cc2ccc(Br)cc2CC1C 70168,C(C(=O)N1OC2CCC1C2)C1CCN(C(C(N=S(C)(C)=O)=O)=O)C1 70169,C1(C2CC2)(NC(C(C)OCCCC)=O)CCN(C(=O)C(C)(C)C(=O)OCC)C1 70170,c1(CC(N2CC3CC(NC(c4c(CC)ocn4)=O)C3C2)=O)c(O)nc(=N)[nH]c1C 70171,C1(CCN(C)C(c2ccc(F)cc2)=O)CCCCN1C(c1n[nH]cc1Cl)=O 70172,c1(CNC(c2c(C)ncnc2)=O)nc(CNC(=O)CN2CCOCC2)cc(O)n1 70173,C(=O)(C1=C(C#N)CCC1)NC1C2C(C(=O)NC(C)CS(C)(=O)=O)C3C(C2)C13 70174,CCS(=O)(=O)CC(=O)NCC1(C(=O)NCC(C)(CO)CO)CC12CCC2 70175,CCCC(CC(C)C)C(=O)NCC1(CNC(=O)C(C)(CC)OC)CCOCC1 70176,C(=O)(C1=CCC(F)(F)CC1)N(C(CNC(C(CC)(F)F)=O)C1CC1)C 70177,C(CCN(C(=O)CC1CC=CCN1C)C)(C(C)(C)C)NC(C1CC(OCC)C1)=O 70178,C1(O)(CNC(C(C)N(C(C2(CCC=C)CC2)=O)C)=O)CCCCCC1 70179,N1(C(C2CCC(CC)O2)=O)CCCN(C(c2cnc(O)cc2C)=O)C(CO)C1 70180,N1(C(c2ccno2)=O)CC(C2CCCN(C(C3(CO)CC3)=O)C2)C1 70181,N1(C(CCOCCN(C(C=C(C)C(F)F)=O)C)=O)CCCC(C)(C#N)C1 70182,CC1C(C(=O)Nc2cccnc2F)CCCN1C(C1CC2(C1)CC2(F)F)=O 70183,C1(C)(NC(C(CSC)O)=O)CCCN(C(c2nc(C(C)C)oc2C)=O)C1 70184,c1(-c2cc(Nc3ncc(OC)cn3)ncc2)ccc(S(C)(=O)=O)cc1C 70185,C1(NC(C(Cn2ccc(C)n2)C)=O)CN(C(c2c[nH]nc2C)=O)CCC1F 70186,C1(C2N(C(C(c3ccncc3)C)=O)CCC2)CCN(C(=O)Cn2cccn2)CC1 70187,c1(COC)cc(C(N2CCOCC2CNC(C2CC2c2cccs2)=O)=O)n(C)c1 70188,C12(NC(C3=NOC(C)C3)=O)CCCC1(F)CN(C(c1ccncc1Cl)=O)C2 70189,N1(C(c2c(CC)occ2)=O)CCC(C)C1CNC(C1OCC1(C)C)=O 70190,C(CC(C(=O)N(C1CCC(CO)CC1)C)NC(C1CC1C(F)(F)F)=O)SC 70191,c1(C(=O)OC)cc(F)c(CO)c(F)c1.C12CN(C(=O)C(F)=CCCF)CC1N2 70192,N1(C(c2c(CC)ccc(Br)c2)=O)CCC(NC(=O)CNC=O)C(C)(C)C1 70193,c1(C(N2CC(C)(OCC(N3C(C)(N(C)C)C=CC3)=O)C2)=O)cc(=O)n(C)cn1 70194,C(CCCC=O)OC(C)=O.CCC(F)(F)CN(CCCSC(=O)N(C)C)C 70195,N1(C(c2ccc(C)cc2OC(F)(F)F)=O)CCC2CCC(C1)N2C(=O)CCC#N 70196,N1(C(Cc2nnc(C)o2)=O)CCN(C(C2CC3(CCC3O)C2)=O)CC2(CC2)C1 70197,N1(C(COCCSC)=O)CCC(C(C)(C)NC(=O)C(O)CSC)CC1 70198,c1(C(=O)NC2(C)CCN(C(=O)CC3CCCO3)C2)cc(S(N)(=O)=O)ccn1 70199,S(=O)(=O)(c1c(F)cc(F)cc1F)N1C2CN(C(c3c(C)nc(C)s3)=O)CC1CC2 70200,N1(C(CC2COCC(C)O2)=O)CCC=C(C(=O)NCCCc2cc[nH]n2)C1 70201,CC1CC(C(=O)NCCc2ccon2)CN(C(=O)Cn2cc(C3CC3)cn2)C1 70202,N1N(Cc2cn(-c3ccc(OC)cc3)nn2)CCOC2(CCOC2)C1 70203,C(CCN=C(NCc1cccc(O)c1)NC1CCCC1)c1c(C)cccc1 70204,c1(-c2cn(C3CN(C(CCOCC)=O)C3)nn2)sc(OC2CCCOC2)nc1Cl 70205,C12(C(=O)NC3C(OCC)CCOC3)COCC1CN(C(C1(C(C)C)CCC1)=O)C2 70206,C1(Cn2cc(-c3n(C)cnc3)nn2)CC2CCC1(NC(c1cc(N)cnc1Cl)=O)C2 70207,C1(CNC(=O)OC(C)(C)C)CCCCCN1C(=O)C(=O)NC(C1CC(C)(C)C1)C 70208,Cc1nccc(C(=O)NC2CC(C(=O)NCCSC(C)C)C23CCC3)c1C 70209,CC(CS(N)(=O)=O)NC(C1(C)CC(NC(C2CC=CC2)=O)C1)=O 70210,C(C(CC1CC1)C(=O)N1CC2CC2(CO)C1)NC(C1CC(=C2CC2)C1)=O 70211,NC(=O)CC(O)C(=O)NC(CNC(=O)CCc1cc(Br)ccc1F)CO 70212,c1(CNC(c2n(C)nc(C)c2Br)c2nnnn2C2CC2)ccc2c(c1)CCCO2 70213,C=CC(C)(O)CC(=O)NCCC1(C(=O)NCC2CCSCC2)CCC1 70214,N1(C(C(CC)NC(C)=O)=O)CC(CNC(=O)C(C)Sc2ncccn2)C(C)C1 70215,c1(C(=O)NCC(C2CCOC2)NC(=O)COC2CCC2)ccc(CO)nc1 70216,CC(CCC(C)(C)C)C(=O)NC1CCN(C(=O)CCc2cnn[nH]2)CC(O)C1 70217,N(C1CCc2cc(Cn3cc(-c4cnc(O)nc4)nn3)ccc21)C(=O)OCC 70218,C=CC(CC)CC(=O)N(CCC(C)NC(=O)CCNC(=O)OCC)C 70219,C1(C(N(CC(=O)O)C(C)C)=O)CCCC(NC(=O)C(C)c2cc[nH]n2)C1 70220,CC1CCCC(C(=O)N(CCc2cccs2)CCNC(=O)OC(C)(C)C)C1 70221,C1(CC(C)NC(C2(C3CC3)CCCO2)=O)CCN(C(c2ccco2)=O)CC1 70222,C#Cc1cccc(C(=O)N(C2CCCN(C(c3n[nH]c(C)n3)=O)CC2)C)c1C 70223,C(CC(C(C)C)NC(=O)C(n1nc(C)cc1C)C)NC(c1cn(CC=C)nc1)=O 70224,C1(NC(CCOCCC)=O)CC(F)CN(C(=O)COCC2CCCOC2)C1 70225,C#Cc1ccc(C(N2CCC(CCNC(=O)CC(C)P(C)(C)=O)C2)=O)c(F)c1 70226,N1(C(c2scnc2C)C(=O)NC)CCC(O)CC12CC2 70227,N1(C(CC2(C)CCCCC2)=O)CCC=C(CNC(c2cccnc2)=O)C1 70228,C(c1cnn(C)c1C)=CC(=O)NCCCOCCCNC(C(C=C)O)=O 70229,c12cccc(c1)C(SC)N2.C1(COC)(SC)CN(C(C)=O)C1 70230,C1(CCOC)CN(C(=O)C(N2CCN(C)CC2)(C)C)CCN1C(c1csnn1)=O 70231,CC(C)(C)C(CNC(C1(F)CCC1)=O)NC(=O)CC(=O)NC1CC1 70232,C1(CC(=O)NCc2ccc(CC)s2)CC(C)N(C(=O)Cc2cnsc2)C1 70233,Cc1cccc(C=CC(=O)NC2CC(O)C2CC(=O)NCC(F)(F)C(N)=O)c1 70234,C1(C(=O)NCC(CC)NC(C2(O)CC2)=O)CC(=O)N(c2ccc(COC)cc2)C1 70235,c1(C(=O)NCC2C3CN(C(C45COC(CCO4)C5)=O)CC23)ccc2cc[nH]c2n1 70236,CC1CC(CNC(=O)CC(C)(F)F)CN1C(c1cnco1)=O 70237,C#CCC(CC#C)C(=O)NCC(CC)(CC)NC(=O)CCC1CC2CCC1C2 70238,N1(C(CCC(=O)NC)=O)CCC2(CCN(C(=O)C(C)OCC3CCCO3)C2)C1 70239,c1(N(C(c2ncc(-c3c[nH]c(=N)c(C)c3)cn2)=O)CC)cccc(O)c1OC 70240,c1(C(=O)NCC2C(NC(c3cn[nH]c3)=O)CCC2)ccc(F)c(Cl)c1F 70241,Cn1ccc(C(=O)NC2CC(CNC(C3CC(C(F)(F)F)C3)=O)C2)c1C1CCC1 70242,CC(C)CC(C(=O)NCc1ccc(CO)o1)N(C(=O)CC(C)C1CC1)C 70243,C(=O)(C(CCC=C(C)C)N(c1ccccc1Cl)C)NCCCSC 70244,N1(C(C(N2CCC(C)CC2)=O)=O)CC(C)N(C(=O)C=C2CCC2)C(C)C1 70245,C1(C(N(C2CN(C(c3c(OC)c(Cl)ncc3)=O)C2)C)=O)Cc2c(F)cccc2O1 70246,C1(NC(c2c(SC)snn2)=O)CN(C(=O)CSCC(N)=O)C2(CCCOC2)C1 70247,C(C1=CCCN(C(C2(C)CCCC2)=O)C1)NC(CCn1ncc(C)c1)=O 70248,Cc1cccc(C)c1NC(=O)C(c1ncc(Cl)s1)N(CC(C)C(C)C)C 70249,c1(C(=O)NC2(c3ccccc3)CCN(C(CC)=O)C2)cc(=O)cc(Cl)[nH]1 70250,c1(C(=O)NCCCCCNC(=O)Cc2ccco2)cc(C2CC2)nnc1O 70251,c1(C(N(CC(O)CN(C)C(C2CCS2(=O)=O)=O)C)=O)cc(F)c(F)cc1Cl 70252,N1(C(c2c(COC)cc[nH]2)=O)CCOCC1CNC(C1CC(F)(F)CS1)=O 70253,c1(COC)cc(=NCC2(O)CCN(C(C3(N(C)C)CC3)=O)CC2)[nH]cn1 70254,c1(C(N2CC(NC(CCOC)=O)CC(C)(C)C2)=O)ccccc1C#CC1CC1 70255,C1(C(N2CC(F)(CNC(c3c(C)sc(C(F)(F)F)n3)=O)C2)=O)COC2(CCC2)C1 70256,c1(C(C)=O)cncc2n[nH]c(C(C)C)c12.N1CC2=C(C1)CN(C(C1(C)CC1F)=O)C2 70257,CCCCCC(O)CC(=O)N1CC(CNC(c2ccccc2-c2ncc[nH]2)=O)C1 70258,N1(CC(=O)N(CC2N(C(C(C)OCC)=O)CCC2)CC)CCNC(=O)C1 70259,CC(CN1CCCCC1)C(=O)NC(C)CCNC(c1nn[nH]c1Cl)=O 70260,c1(CN(C)C(CCCCNS(C)(=O)=O)=O)ccc2cnccc2c1 70261,C#CC1(CNC(C2CC(CNC(=O)CNC(=O)C3CC3)C2)=O)CC1 70262,c1(C(N2CC(C)C(NCc3ccc(F)cc3F)C2)=O)cccc2c1CCC(=O)N2 70263,C1(NC(COC)=O)CCCC(NC(=O)OCCC(=O)N(CC(C)C)C(C)C)C1 70264,c1(CC(N2CC(CCNC(C3CC(CC4CC4)C3)=O)(OC)C2)=O)ccccc1F 70265,N1(C(C2CCCN(CC)C2)=O)CC2(CC(CC(=O)NC3(CCF)CC3)C2)C1 70266,N1(C(C2N(C)S(=O)(=O)CC2)=O)CCCC2(CCCN2C(C2CC(O)C2)=O)C1 70267,c1(C(N2C3C(NC(c4n(CC#C)ccc4)=O)C(CC3)C2)=O)ccc2nonc2c1 70268,N1(C(C=Cc2ccc(C(=O)OC)o2)=O)CCCC(C2CN(C(=O)C(C)O)C2)C1 70269,C(=O)(CCC(C)(C)NC(c1nnnn1CC(F)F)c1ccno1)OC 70270,C1(=CC(N2CC(CNC(CCc3ncc(C)[nH]3)=O)C3C2C3)=O)CCCCC1(C)C 70271,C(=O)(C(F)C(F)(F)F)N(CC1OCCN(C(C2C(C(C)=O)C2(C)C)=O)C1)C(C)C 70272,N1(C(C(C)CC(F)(F)F)=O)CC2(C)CN(C(C3CC4(C3)CC(O)C4)=O)CC2(C)C1 70273,N1(C(c2cn(CC(=O)N(C)C)nn2)=O)CC2CC2(CNC(=O)C(F)(F)C2CC2)C1 70274,N1(C(c2c(C)cc(C)c(C)c2)=O)CCC2CCN(C(=O)CSCCC#N)CC12 70275,C1(F)(C(=O)NC(C(C)C)CCN(C(=O)C=Cc2nnn(C)n2)C)CC2(CCC2)C1 70276,c1(NC(c2ccc(OC)c(OC)c2)C#N)cccc2c1OCCC2O 70277,N1(C(c2n(CC)cc(Cl)c2)=O)CCC(O)C(NC(C2CC3(CCCO3)C2)=O)C1 70278,CCCC(O)C(CO)NC(=O)C1=NOC(CNC(C2CC3(CC3)C2)=O)C1 70279,C1(C(=O)NC2CCCCCC2)CC2(CCC2)CN1C(c1ccccc1O)=O 70280,c1(CN2CCC(C(C)=O)C2)cccc(Cn2nc(C)cc2C)c1 70281,C(=O)(C(C(C)C)NC(=O)COC1CC(n2cc(COC3CCCC3)nn2)C1)OC 70282,C12(CNC(C(C)OCCCCCC)=O)CC(CN1C(=O)C(O)Cc1cnc[nH]1)C2 70283,N1(C(CC(=O)NCC#C)=O)CCC(C)C(NC(=O)C(CC)n2cccn2)C1C 70284,C=CC1CN(C(C2CC3CC3C2)=O)CC1NC(=O)CCOCC(F)(F)F 70285,c1(C2N(C(c3c(OC)oc(C)n3)=O)CCC2)cccc(Cl)c1Cl 70286,C1(NC(CC)=O)CCN(C(=O)Cn2nccn2)C1Cc1ccccc1 70287,c1(N2CCN(C(=O)NOCCc3cccs3)CC2)ncnc2ccccc12 70288,C(=O)(C=C=C(C)C)N1C(C(=O)NCCC2(COC)CC2)CC1C 70289,CCCC(C(=O)OC)C(=O)N1CCN(C(c2cnco2)=O)CC1COC 70290,N1(C(Cn2c(CCC)ncc2)=O)CCC(O)C(N(C(=O)C(F)C2CCC2)C)C1 70291,Cc1cc(O)cc(O)c1CNCC1CCCCN(C(=O)C(F)F)C1 70292,C#CC1CCC(C(N2CCOC(C(C)NC(=O)COc3cn[nH]c3)C2)=O)CC1 70293,c1(C(C(N2CCC(O)(CNC(c3ncccn3)=O)C2)=O)O)ccc(F)c(F)c1F 70294,C(=O)(C1CC(=O)Nc2cc(F)ccc21)N1CC(NC(c2n(C)ncc2)=O)C2C1C2 70295,C(C(C)(O)C(=O)NCc1cccc(F)c1)OC.C12CC(C1)NC(=O)CCNC2=O 70296,CCC(C)(C)C(=O)C(=O)NC1(CO)CCCN(C(=O)C(c2ccc(C)cc2)O)C1 70297,c1(C(=O)NCC2(C)CCCN2C(C2CC(CF)C2)=O)cccn2cnnc12 70298,CC(CC(F)(F)F)C(=O)NC12CCC(CC1NC(c1cn3ccnc3s1)=O)C2 70299,c1(C(=O)NC(C(C)NC(c2cnn(C(C)(C)C)c2)=O)C)cc(Cl)n(C)n1 70300,C1(NC2(c3ccccc3)CC(F)C(F)(F)C2)Cc2nc3ccccc3n2C1 70301,C1(CCC(C)C)CCN(CC(=O)NCCC2CCCCC2)CC1 70302,c1(CNC2CC3(N(C(CCCCC(=O)OC)=O)CC3)C2)cccc2cnccc12 70303,c1(OC(C(=O)NCC2CN(C(CC3C(C)C3)=O)C2)C)cccc(Br)c1 70304,Cc1cc(C=CC(N2CCN(C(=O)C(C(C)C)N(C)C)CC2C)=O)c[nH]c1=N 70305,C1(C(N(C)CC2N(C(c3cc(C)c(C)o3)=O)CCC2)=O)CCC2C(CC1)C2(F)F 70306,Nc1sc2c(c1C(N1CC(O)(CNC(C3C4CCCC34)=O)C1)=O)CCC2 70307,CCC(CNC(C12CC(C)(C1)C2)=O)(CC)NC(=O)CCn1cccn1 70308,C(=O)(CS(=O)(=O)CC(C)C)NCC1CCN(c2snc(SC)n2)CC1O 70309,C1(CC(=O)NC2(C)CC(C(=O)OC)C2)CN(C(=O)CCC2OCCO2)CC1C 70310,c1(C(N2CCOCC(NC(C)=O)C2)=O)cnc2[nH]ncc2c1 70311,C1(OC)(CNC(=O)CC2(C)CCN2C(=O)C(C)OCC(C)C)CCOC1 70312,N1(C(C2C(C)=C2)=O)CCC2(CCOCC2)C(NC(c2cc(CO)nc(Cl)c2)=O)C1 70313,C1(C(=O)NCC2CC(NC(c3ccnnc3O)=O)C2)OCC2CCCCC12 70314,C1(COC(C2CCS(=O)CC2)=O)CCCC(C(F)(F)F)C1 70315,Cc1ncsc1C=CC(N1CC2C(CNC(c3ccc[nH]3)=O)C2C1)=O 70316,C1(CNC(CCC2CCC(=O)N2)=O)CC2(CC2)CN1C(c1nc(Cl)c(Cl)s1)=O 70317,C(=O)(C(F)(CNC(=O)C(CCC)N(C)C)C(C)C)NCCCCCC 70318,C1(C)(CC(=O)NCCN(C)C2CC2)CCN1C(=O)CC1CC(F)(F)C1 70319,c1(C(=O)NCCCCN(CCCNC(C(C=C)O)=O)C)c[nH]cc(C)c1=O 70320,Cc1cc(CC=O)cs1.C(=O)(CSC(C)(C)C)N(C)CCNC 70321,c1(C(C)=O)cc(Cl)ccc1C(N1CCC(c2ccc(OC(F)F)cc2)C1)=O 70322,N1(C(c2ccc(C)cc2F)=O)CCC2(CCC(CC(=O)NC(C)C#N)CC2)CC1 70323,N1(C(c2cc(C(=O)Nc3ccc(C)cc3OC)no2)=O)CCC(COC)C(O)C1 70324,c1(C(C)C)ccc(OCCCC(=O)NC(C)CN(C)C(C2CSC2)=O)cc1 70325,C=CCCCCCC(=O)N1CCN(C(c2ccc(C(F)(F)F)nn2)=O)C(C)C1C 70326,CCS(=O)CC(=O)NC1CC1NC(c1ccc(NC(=O)NC2CC2)nc1)=O 70327,C1(C2CCN(CC(=O)NC(CC)(C)C)C2)CCCCN1C(=O)CN1CCOCC1 70328,C(=O)(CC(CC(N)=O)c1ccc(F)cc1)N(CCCNC(C1COC(=O)O1)=O)C 70329,c1(C(N2CCC(OCCNC(C3C(C)CCC3)=O)CC2)=O)ccnc2c1CCO2 70330,c1(C(=O)NCC2OCCN(C(c3cc(C(C)C)[nH]n3)=O)C2)ncccc1N=[N+]=[N-] 70331,C1(C(N(CCCCNC(CCCC(C)C)=O)C)=O)CCc2n[nH]cc2C1 70332,c1(CCCC(=O)NCC(C)N(C(C(C)OCC2CC2)=O)C)cccc(Cl)c1 70333,C1(C(N(C2CCCN(CC3CCOCC3)CC2)C)=O)CC2CC2CC1C 70334,C(=O)(C(O)CC(F)(F)F)N1C(c2cn(C3C(C)(C)CCCC3)nn2)CC1 70335,CCC(C)CCCCC(=O)NC1CC(C)N(C(c2ccc3oc(O)nc3n2)=O)C1 70336,C(c1ccc(OC)c(F)c1)=CC(=O)NCC(C(=O)OC)CC1CCCC1 70337,c1(C(C)NC(C2(C(C)NC(=O)OC(C)(C)C)CC2)=O)ccc2ccn(C)c2c1 70338,O=S(=O)(c1cc(F)cc(F)c1)Nc1ccc(Br)c(Cl)c1F 70339,c1(C(N2CC(COC)(NC(c3ccc(=NC)[nH]c3)=O)C2)=O)ccn2nnnc2c1 70340,C1(C(N(CCN(CC(COCCOC)O)C)C)=O)(OC)CCCCC1 70341,C1(NC(c2cccc(OC)c2)=O)C2CCC1CN(C(C1CCC(=O)N1)=O)C2 70342,C=C1CCN(C(=O)CC2CC2(C)C)C(C(=O)NC2CNC(=O)C2(C)C)C1 70343,c1(C(C)OC)nc(-c2c[nH]ccc2=O)n(CC2CCCOC2)n1 70344,C(C(=O)NCCN1CCN(C(=O)C(=O)NCCC(N)=O)CC1)(C(C)(C)C)OC 70345,Cc1ncc(NC(C2(CCC3CC3)CCC2)=O)c(C)c1C.C12(CC1)C(=O)NC2=O 70346,c1(C(=O)NCC23CC(NC(CC4C(C)CCO4)=O)(C2)C3)c(Cl)csc1Cl 70347,CN1CCCCC1C(=O)NC1(CNC(c2cccc(C3(C#N)CC3)c2)=O)CC1 70348,CC(C)CC(C(=O)N1C2CCCC1CC(NC(=O)Cc1cn(C)cn1)C2)C(C)C 70349,C1(C(=O)NCC(C)N(C(c2ccc(F)cc2F)=O)CC)CN(CP(C)(C)=O)C1 70350,N1(C(C(C)=CC)=O)C2CCC1C(CNC(=O)CCC(=O)NCc1ccccc1)C2 70351,c1(C(C)NC(=O)NC(C(=O)OC)C)cccc(F)c1 70352,C(C(CC(=O)NC(C(C)C)C(C)C)C1CCC1)NC(C1C(CSC)CC1)=O 70353,C#CCCCCCC(=O)NCc1cc(C(=O)NCC(C)C(C)CC)n[nH]1 70354,CCCCCC(O)CC(=O)NCC1CCCN1C(c1cnn(C)c1C(C)(F)F)=O 70355,C(CC1CC1)(CC(=O)NCC1CC1c1ccoc1)NC(C=C(CCC)C)=O 70356,CCC(CC(=O)NC1COCCOC1)NC(=O)C(C)C1(O)CCC1 70357,C#CCCC(C(=O)N(C(CO)C(C)C)C)NC(=O)C(C)SC(C)C 70358,C1(C(=O)NCCC(=O)NC(CC)C)CCN(C(C2CC2Cl)=O)C12CC2 70359,C1(C(=O)NCC=CCNC(C2(CC=C)CCCC2)=O)Cc2nnc(C)n2C1 70360,C1(NC(CCOCC(C)C)=O)CCC(C(N2CCC2CC2CC2)=O)C1 70361,c1(C(N(CCN(C(=O)CCC(C)O)C(C)C)C)=O)cc2n(n1)CCCC2O 70362,C1(NC(=O)C2=CCCOC2)CCN(C(=O)CC2CC3CC3C2)CC12CCC2 70363,c1(-c2cncc(NS(CCOC)(=O)=O)c2)ccc(F)c(NCC2CCCCO2)c1 70364,c1(C(N2CC(NC(c3cn(CCC)nc3C)=O)C2)=O)ccc([N+](=O)[O-])cc1F 70365,C12(C(=O)NCC(=C)CCNC(C3NC(=O)OC3C)=O)CCCCC(=O)N1CCC2 70366,N1(C(C(CC)n2nccc2C)=O)CCC(NC(c2cnc(C)cn2)=O)C(C)(C)C1 70367,Cc1cc(C(N2CC3CC(NC(c4nnc(O)cc4O)=O)C2C3)=O)c(C)cc1Cl 70368,C1(NC(C2CC(OCC)C2)=O)CCC(CNC(=O)CSc2nnnn2C)C1 70369,N1(C(C(C)c2cc[nH]n2)=O)CC(CNC(c2cc(C(N)=O)no2)=O)C2(CC2)C1 70370,C1(C)(C(N2CCC(CCOC)C2)=O)CCN(C(=O)C(C)CC(N)=O)CC1 70371,C12(CC(=O)NCCOCC)CCC1CN(C(=O)CCc1cccn1C)C2 70372,c1(C(N2CC(C)C(CNC(C3CC(C)(O)C3)=O)CC2)=O)ccc2c(c1)CCC=C2 70373,CC#CCC(C(=O)N(CCS(N)(=O)=O)C)NC(C1CC(SC)C1)=O 70374,c1(C(=O)NC(C(C)NC(Cc2cc(C)[nH]n2)=O)C)c(C)ccnc1O 70375,C1(CNC(CC(C(=C)C)OCC)=O)CC2CCC1N(C(C1(Cl)CC1)=O)C2 70376,c1(C(=O)NC2(COC)CN(C(=O)C(C)SC(C)C)C2)cccc2ccsc12 70377,N1(S(CC)(=O)=O)CCC2(CC(C(=O)Nc3cccc4c(O)cccc34)=NO2)C1 70378,C1(NC(=O)NC2CCN(C(C)C)CC2)CC2CC(Nc3ccc(F)c(F)c3)CC12 70379,N1(C(CC(COC)C)=O)CCC2(CCCN2C(=O)CCc2nc(=N)[nH][nH]2)CC1 70380,c1(C(N(CCNC(CC2(COC)CC2)=O)C2CC2)=O)cnc2ncnc(O)c2c1 70381,C(=O)(C1CCCn2nccc21)N1CC(O)(C(CNC(C(C)C#N)=O)(C)C)C1 70382,N1(C(C(=O)NCCCCCC)CCC2CCCO2)CCCC(CCO)CC1 70383,Cc1nc(N(C2C3CCOC3C2(C)C)C)c2sccc2n1 70384,Cc1ccc(F)c(C(=O)NC(Cc2ccoc2)C(=O)NCc2ccc[n+]([O-])c2)n1 70385,C12(NC(CCSC)=O)CN(C(c3nc(C)n(C)c3C)=O)C(COC)(C1)C2 70386,c1(C(=O)NC2C(NC(C3CCCC(C(=O)OC)C3)=O)CCC2)cn2nc(C)sc2n1 70387,N1(C(C(C)=C2CCCC2)=O)CCC(CNC(C2CCCN2CC(F)(F)F)=O)C1 70388,C1(C(N2CC3C(CNC(C4CCCC4)=O)(C3)C2)=O)CCN(CCO)C(=O)C1 70389,CCC(CC(=O)N1CC2C(C(=O)NCC(C)(C)CN=[N+]=[N-])C2C1)C(F)F 70390,CCCCCCCCCC(=O)NCC1CN(C(=O)C2=NNC(=O)CC2)CCO1 70391,c1(N2CCCC(CCCCCC)C2)nc(=N)[nH]c(=NCc2nocc2COC)[nH]1 70392,C(C(COC)CC(=O)NCCCC(=O)NCC1COCC1O)OC 70393,c1(C(=O)NC(CC)CN(C(=O)C(O)C2CCCC2)C)ncn(-c2ccccc2)n1 70394,C1(C(N2CCC(CO)(CNC(=O)C3=CCSC3)C2)=O)(OC)CCCOC1 70395,C(=O)(C(C)(C)C(C)O)N1CCCC(CN(C(c2c(C)oc(Cl)n2)=O)C)C1 70396,c1(C(N2C(C)CC(NC(c3ncc(OCC)nc3)=O)C2)=O)cc(C)nc(Cl)c1N 70397,Cc1nc(C(N2CCCC2C=CC(=O)NC2(CN(C)C)CCC2)=O)sc1C 70398,C1(C2CC2)(C(=O)NC2CC(CCNC(C34C=CC(CC3)C4)=O)C2)CCOCC1 70399,c1(CC(=O)NC(CC)(CNC(c2ccn(C)n2)=O)CC)cccc2c1OCO2 70400,Cc1ccc(F)c(C(=O)NC2CC3CC2CC32CC2)c1Cl 70401,C1(CNC(C(C=C)O)=O)CCCC2CN(C(=O)CCCCC(=O)NC)CC12 70402,c1(C(N2C(CNC(CC(CCC)(C)O)=O)CC2)=O)cc(F)cc2nccnc12 70403,C1(NC(c2c(C)cc(C)[nH]2)=O)CS(=O)(=O)CC1NC(=O)CCC1CCCCC1 70404,C#CCC(C(=O)NC)NC(C1(C)CCN(C(=O)C=C(C)C(F)F)C1)=O 70405,C1(CS(N2CC(C)(N(CC)CC)C2)(=O)=O)C(C)CCCC1C 70406,C(=O)(C(O)C(F)(F)F)NC1CCC(CC(=O)N(CC)Cc2ccncc2)C1 70407,c1(C(N(C(CN(C(C(COCC)C)=O)C)C)C)=O)cc2n(n1)CCCC2 70408,N1(C(c2cc(C)oc2)=O)CCC2CN(C(C3CC4C(C3)C4(F)F)=O)CC12 70409,C(CN=c1[nH]c(Cl)ncc1C)C1CC(NC(C2(CC)CCNC2=O)=O)C1 70410,C=CCC(C(=O)NC1CCCCC1CNC(c1c[nH]nc1Br)=O)C(C)C 70411,c1(C(N(CCCNC(C2CC(O)(C(F)(F)F)C2)=O)C)=O)ncn2c1CCCC2 70412,C1(NC(CCc2cnc(C)nc2O)=O)CN(C(=O)Cn2ncnn2)CC1C1CC1 70413,N1(c2ncnc3[nH]cc(I)c32)CCC(C2CN(Cc3cnc(C4CC4)s3)C2)CC1 70414,N1(C(=O)C(F)C2CC2)CCN(C(=O)CCCn2ccnn2)C(CC2CCOCC2)C1 70415,Cc1cc(C(=O)NC2CN(C(c3cc(O)no3)=O)CCC2C(F)(F)F)cnc1F 70416,N1(C(=O)CC2(O)CC2)CCC2C(C1)CN2C(C1CCOCC1)=O 70417,c1(CC(=O)NC2CCCC(NC(COCCC#C)=O)C2)noc2ccc(F)cc12 70418,Cc1nc(C(N2CCC(C(C)NC(=O)CCCc3cccnc3)C2)=O)c(C)s1 70419,N1(C(c2c(F)cccc2Cl)=O)CCC2C(CCN2C(=O)CCn2cncn2)C1 70420,C=CCC(C)C(=O)NC1CCC(N(C(=O)CC2C(=O)NN=C2C)CC)CC1 70421,c1(C(N2CC(COC)(NC(C3C4CCCC34)=O)C2)=O)ccc(Cl)cn1 70422,C1(C2CC2)(CNC(c2c(C(C)C)ccs2)=O)CCN(C(=O)C(O)C2CCC2)C1 70423,N1(C(C23N(C(CN(C)C)=O)CCC2CCC3)=O)CCC2(CCCCC2)C1 70424,c1(CC(N2CC(C(C(=O)NC(c3nccs3)CC)O)C2)=O)cncnc1 70425,C1(C(C)NC(=O)C=Cc2cc[nH]c2)CCCN(C(C2(C(F)F)CCCCC2)=O)C1 70426,CC1C(=O)NC(=O)CN1C(C1(C)CN(C(c2cc(=N)[nH][nH]2)=O)C(C)(C)C1)=O 70427,C(C(CO)C(F)(F)F)NC(C(CC1CC1)NC(c1nn(C)c(O)c1)=O)=O 70428,CCC(CO)C(=O)NC(C)CC(C)NC(C1(NC(C)=O)CCCC1)=O 70429,C1(CC)CCN(C(C2CC23CCC3)=O)C1C(=O)NCC(=O)NC(C)(C)C 70430,CC(CC=Cc1ccccc1)C(=O)N1CCC(NC(C2OCCO2)=O)C1 70431,C(C)(CCCC(=O)NCC1OCC2CCC1C2)NC(C(C)NC(CC)=O)=O 70432,C12(NC(CN=S(C)(C)=O)=O)CCOCC1CN(C(c1ccncc1)=O)C2 70433,C(=O)(C1CCCn2ccnc21)N1CCCC(O)(CNC(CCCS(N)(=O)=O)=O)C1 70434,c1(C(=O)NCCOCCN(C)C(C2(C)CCNC2=O)=O)ccc2c(n1)CCO2 70435,C(N=c1nc(OC)c2nc[nH]c2[nH]1)C1CCN(C(C2(CSC)CC2)=O)C1 70436,C(c1ccc(C(=O)N(CCCNC(=O)C(F)CC2CCCC2)C)o1)=CC(=O)OC 70437,CC(CNC(C1(C)CCN(C)C1)=O)CC(=O)NCCCC(F)(F)F 70438,C1(NC(CCC(=O)NC)=O)CC(O)CN(C(=O)CCCNC(N)=O)C1 70439,c1(C(=O)NC2C(N(C(=O)CCC3CCOC3)C)CCCC2)cccc2nc[nH]c12 70440,C=C(Cl)CC(C(=O)NCCCC(N)=O)NC(c1coc(SC)c1)=O 70441,C1(CCC(=O)N(C2CC(C)C2)C)CCCCN(C(C2(O)CCOC2(C)C)=O)C1 70442,C1(NC(CC2(NC(C)=O)CC2)=O)CC2C(NC(=O)C(c3ccccc3)C)C2C1 70443,N1(C(C(CC)NC)=O)CC2CN(C(c3cnc(Cl)c(C)c3)=O)CC12 70444,Cn1nnc2c1NC(C(=O)NCCC1CC3CCC1C3)CC2 70445,N1(C(C(CCC)(C)O)=O)C2CCC1C(C)C(NC(C1CCC(C(N)=O)CC1)=O)C2 70446,c1(NC(N2CC(CCN3CCOC3=O)C2)=O)cc(Cl)ccc1I 70447,N1(CC)CCCCC1C(=O)NCCCC(=O)N(CCCC(C)O)C 70448,CC(C)CC(CNC(C1CC2CC2N1C(C12CCC(CC1=O)C2)=O)=O)CO 70449,C1(NC(=O)Cc2cc(C(F)(F)F)n[nH]2)CC1C1CCCN(C(=O)C=CI)C1 70450,C1(CNC(C(=O)NCC)=O)CN(C(c2cn(C3CCOC3)nn2)=O)C(C)(C)C1 70451,C(=O)(CS(=O)(=O)c1ccccc1F)N1CCC(CC=C)(NC(=O)CC=C(C)C)C1 70452,CCCC(O)C(=O)NCCC1CN(C(=O)C(F)(F)c2cccnc2)CC1C 70453,Nc1cc(C(=O)NCCOC2CN(C(=O)CCc3ccncn3)C2)cc(Cl)n1 70454,C1(C(=O)NCC2C(C)(C)CCN2)Cc2ccc(O)cc2CN1 70455,C#CCC(CC#C)C(=O)N1CC2CCC1C(CNC(=O)CC(CN(C)C)CC)C2 70456,c1(C(=O)NCCN(CC(=O)NC2CC2)C2CC2)ccoc1I 70457,c1(CN2CCN(C3CCN(C(C4CC5(CC5)CO4)=O)C3)CC2)cc(Cl)cc(Cl)c1 70458,C12(CC)CCC(C(=O)NC3CC3CNC(=O)CCc3ccc(F)c(F)c3)(CO1)C2 70459,c1(C(N2C(CCCNC(CN(C(C)=O)C)=O)CCC2)=O)cc(C(F)F)ccn1 70460,C#Cc1ccc(F)cc1C(=O)NC1CN(C(=O)CC(C)F)CC1n1cccn1 70461,C(=O)(C(C)C(CC)CC)N1C(C(N(CC(=C)C)C)=O)CC(=O)C1 70462,c1(C(=O)NC2(CNC(c3n(C=C)ncc3)=O)CCOC2)cc2sc(Cl)cc2s1 70463,C(CNC(c1cnc(C#N)s1)=O)(C(C)(C)C)NC(C1(COC)CC1)=O 70464,C=C(C)C(C)(C)C(=O)NCC1CN(C(=O)C(C2CC2)OC)CCC1C(F)(F)F 70465,c1(C(N2CCCC(N(C(CCC#CC)=O)CC)C2)=O)ccc2ccnc(Cl)c2n1 70466,c1(C(N2CCN(C(c3c(OC)c(Cl)sc3)=O)CC2)=O)n[nH]c2c1CCC2 70467,C#CCC(C)(C)C(=O)N1CC(C(=O)Nc2cncc(N(C)C)c2)C(C(C)C)C1 70468,C(=O)(CCCCCN(C)C)NC(C)CC(N1CCC(C#N)C1)=O 70469,C1(C(=O)NC2C(NC(c3c(Cl)cn(CCC)n3)=O)CCC2)CCc2nncn2C1 70470,C1(CC(=O)NC2CCN(C(c3ccoc3)=O)C2)CC(C2CC2)C1.C1CC(=O)N1C 70471,c1(C(=O)NC2(C)CC(NC(CC(=C=C)C)=O)C2)cc[nH]c2nccc1-2 70472,CC(C)C1=NOC(C(N2CCC(C(C)NC(C3CC(=O)C3)=O)C2)=O)C1 70473,C=C=CCCC(=O)NCCC1CCC(NC(=O)CCS(C)=O)C1 70474,C1(NC(C2CCC(C(=O)OC)CC2)=O)CN(C(=O)C2=CCCC2)CC1C#N 70475,C1(NC(C=CC(C)(C)SC)=O)CCCC1NC(=O)C(C)CC1CC1 70476,N1(C(c2cc(C)ncc2)=O)CCC2CC2(C(N2CCC(OC(C)C)CC2)=O)CC1 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70494,N1(C(C(CC(C)C)N(C)C)=O)CCC2(CC(C(N3CC(O)CC3(C)C)=O)C2)C1 70495,N1(C(c2cncc(NC)c2)=O)CC(O)C(O)C1CNC(C1CC1OC)=O 70496,N1(C(C=CC)=O)CCN(C(C2CC3CC23)=O)CC1 70497,C(=O)(C(C(C)(C)C)N(C)C)N(C)CC1CCN(C(c2c(COC)ncs2)=O)C1 70498,C(=O)(C(CO)C(C)(C)C)N1C(c2n(C)ncc2)CN(C(=O)CNC=O)CC1 70499,CCCCS(=O)(=O)NC(C(=O)N1CC(CO)(NC(=O)C(C)CF)C1)C(C)C 70500,C1(C(=O)NCCCCCCN(C(CCC(C)OC)=O)C)CCCN2CCCCC12 70501,c1(CCC)ccc(C(N2CC(NC(=O)C(F)F)CCC2C)=O)cc1S(N)(=O)=O 70502,C1(C(=O)NCCOC2CN(C(CCc3cnc(C)s3)=O)C2)CN(C)CCO1 70503,C=CCC(F)(F)CNC(C1(CO)CCN(C(c2ccc(CC)[nH]2)=O)C1)=O 70504,N1(C(C2C(C)CCC2)=O)CC2CN2N=CC(C(N2CC(S(C)(=O)=O)C2)=O)=CC1 70505,Cc1cc(CC(=O)NC2(C(=O)NC(CO)C(C)C)CC2)nn1C 70506,c1(C(N2CC(CNC(c3c(OC)ccs3)=O)C(C)(C)C2)=O)ccc2snnc2c1 70507,CN(C)NC(=O)CCC(=O)Nc1ccn(CC2CCC(F)(F)CC2)n1 70508,CC1(C)CNCC1OCC(=O)NCCC(c1ccccc1)CO 70509,C1(NC(c2c(C)cc(CNC(C(C)=CC3CC3)=O)o2)=O)CCCC1C1CC1 70510,C1(CSC)CCCN(C(n2nnnc2C)C(=O)Nc2ccccc2)CC1 70511,c1(C(N2C(CCNC(C3(CC#C)CCCO3)=O)CCCC2)=O)cnc(F)c(Cl)c1 70512,c1(NC(C2CCN(Cc3c(CC)cccc3)C2)=O)cc(F)c(F)cc1Cl 70513,c1(CN(C(=O)C(N2CCCCC2c2nnc(C)o2)=O)CCOC)ccc(F)cc1F 70514,C1(NCCCNC(N(CCCC#C)CC)=O)CCN2CCCC2C1 70515,C(=O)(CC(C)C(F)F)N(C1CN(C(c2nc(C)oc2C)=O)CC1O)C 70516,Cc1cc(C(=O)NC2CCCCC2NC(c2cccs2)=O)nn1CC(F)(F)F 70517,c1(C(N2CC(CC=C)(NC(c3csc(C(C)C)n3)=O)C2)=O)cnc(C)c(C#N)c1 70518,C1(CC)CCN(C(C2CCC2COC)=O)C(C(=O)NC2C(O)CC2O)C1 70519,n1(CC(N2CC(CNC(COc3cccc(C)c3)=O)C2)=O)cc(P(C)(C)=O)cn1 70520,c1(CC)c(C(N2CCN(C(=O)Cc3cc(C4CC4)no3)C3CC23)=O)cccc1C 70521,N1(C(C2(C#N)CCSCC2)=O)C2CCC1CN(C(C1Cc3ccccc3S1)=O)C2 70522,CC1(C)OC2CC(C(=O)NC3(CNC(C4OCC5CCCCC45)=O)CC3)CC2O1 70523,Cc1ccc(-c2cnc(NC(=O)C(C)NC=O)c(O)c2)c(C)n1 70524,n1(CC(=O)NC2CC(NC(CC3C(C)=NOC3=O)=O)C(O)C2)ccc(O)nc1=O 70525,c1(OC)ccc(Cl)c(CC(=O)NC2CC(NC(=O)C=C(Cl)Cl)C23CCC3)c1 70526,C1(C(N2CC=C(CNC(c3cc(=O)cc[nH]3)=O)CC2)=O)CC1C1CCCCC1 70527,N1(C(C(CC#C)O)=O)CCC(C2CCC2)(CNC(=O)C(C(C)C)OC)CC1 70528,C1(CNC(c2ccc(C(F)(F)F)[nH]2)=O)CN(C(C2CSC2)=O)C2CC12 70529,N1(C(c2c(N)ccc(Cl)c2)=O)CCCN(C(C2(CO)CC2(F)F)=O)CC1CO 70530,c1(OC(C)C)cccc(C(=O)NCC(CO)NC(c2cc(O)cs2)=O)n1 70531,CC(O)C(F)(F)C(=O)NC1CC(F)(CNC(=O)C(c2ccccc2F)(C)C)C1 70532,C1(CC(=O)N(C(C)CNC(C2CCC(N(C)C)CC2)=O)CC)CCS(=O)(=O)C1 70533,c1(C(N(C)CC2CC(F)CN2C(c2ccsc2)=O)=O)cn(C)cc1C(F)(F)F 70534,c1(C(N(CCOCCC(N2CC(=CCC)C2)=O)C)=O)ccc(F)cc1F 70535,Cc1cc(CC(=O)NC2CCCC(NC(=O)CCOCC(C)C)C2)cc(C)c1 70536,c1(CCC)nc(C)c(C(N2CCC(NC(C3CC3C)=O)C2C)=O)s1 70537,c1(C(=O)OCC2CC3(CCC3)C2)ccc([N+](=O)[O-])c(O)c1 70538,Cc1c(Br)ccc(O)c1C(=O)N(C)CC1CCCN1C(C1(C)C=CCC1)=O 70539,C1(CC)CC(C(N2CCC(F)(CNC(c3cc(F)n(C)n3)=O)C2)=O)CC(=O)N1 70540,O=C(C(O)Cc1ccccc1)NC1CC(F)(CNC(c2nsnc2O)=O)C1 70541,C1(C)(CNC(C2(OC)CC2)=O)CCC(NC(c2cc(CCO)on2)=O)C1 70542,C(=O)(CCS(C)=O)N1CC(C(C)NC(=O)C(C)(C)N2CCOCC2)C1 70543,C1(NC(=O)CC2CCCC2)CCCC12CCN(C(=O)CC1CC3(CC3)CO1)CC2 70544,C1(NC(c2cc(O)nc(C3CC3)n2)=O)CC2CN(c3ncc(F)cn3)CC2C1 70545,N1(C(CNC(=O)NC)=O)CCN(C(=O)CC(C)(C)C2CC2)C(C(F)F)C1 70546,C1(CNC(CCN(C)C)=O)(NC(=O)COC2CCCCC2)CCOC1 70547,C1(CNCC(=O)OCCOCCOCCOC)CCCCN1C 70548,N1(C(=O)C=Cc2ccco2)CC23CCCC2(C1)CN(C(c1cc[n+]([O-])cc1)=O)C3 70549,C1(NC(C2(F)C(C)C2)=O)CCC(C)N(C(=O)Cc2ccc(C(F)F)cc2)C1 70550,CC(C)C(C)C(CNC(=O)CCN1CCCC1)NC(c1ccc(CO)cc1F)=O 70551,c1(SC)cc(C)ccc1C(=O)NCC1(O)CCN(C(c2nn(C)cc2C)=O)C1 70552,C1(CNC(C2CN(C(C)=O)C2)=O)CC(NC(c2n[nH]cc2Br)=O)C1(C)C 70553,c1(CN2CC(CC(N3CCS(=O)(=O)CC3)=O)C2)ncccc1[N+](=O)[O-] 70554,C(C1c2ccccc2CCN1C(c1ccc(C(N)=O)c(Cl)c1)=O)NC(C(C)C)=O 70555,c1(OC)cccnc1CN1CCCC(C(=O)NCCCN2CCCC2)C1 70556,c1(C(=O)NCCCN(C(c2cc(CCC)on2)=O)CCC)ccncc1OC 70557,N1(Cc2cn(CCC(C(=O)OCC)C)nn2)CCC12CCSCC2 70558,C1(NC(c2ccc(S)cc2)=O)CN(S(=O)(=O)c2cccs2)CC1(F)F 70559,c1(SC)ccc(C)c(C(N2CCC(C)(CNC(=O)C(O)P(C)(C)=O)C2)=O)c1 70560,c1(N(C(=O)CC2CCN(C(=O)Cn3cnnn3)CC2)C)ccccc1Cl 70561,C1(C(=O)NCC2CCN2C(=O)CSC(F)(F)F)CCCC1C(F)(F)F 70562,c1(C(N2CC(C(C)(C)O)(CNC(=O)CNC=O)C2)=O)cc2n(n1)CC(F)C2 70563,CC1CC(c2nnnn2CC2CCOC2)(NCC(C)(C)CO)CC(C)O1 70564,N1(C(c2c(C)n(C)cn2)=O)CC(C(=O)NCc2cnn(C)c2O)CC1(C)C 70565,C(C#Cc1cccnc1)NC(C1CCCN1C(c1cccn2cncc12)=O)=O 70566,N1(C(C(=O)NCCN(C(C2CC(OC)C2)=O)CC)C)CCCC(O)C1 70567,c1(CC(=O)N(CC(CNC(CC2CC(OCC)C2)=O)C)C)cc(C)on1 70568,N=c1ncn(CC(=O)NCCOCCNC(C2(CF)CC2(F)F)=O)[nH]1 70569,C(C1=CCN(C(C2CCCS(=O)(=O)C2)=O)CC1)NC(C1CCC(C)O1)=O 70570,N1(C(=O)OC(C)(C)C)CCC(C(=O)N(C2CCC2)CC2CC2)C1 70571,C1(C)(C(N2CCC(OOCC(=O)NCC3(CC)CC3)C2)=O)CCC2CC2C1 70572,C1(C(=O)NC(CCC)C2CCC2)CCN(C(C2C=C(C)CS2)=O)C(C)(C)C1 70573,N1(CCN(C)C(C2CCOC(=O)CC2)=O)CCSC(C)(C)C1.C12CN(CCO1)C2 70574,C1(Cn2cc(-c3c(C)nsc3)nn2)CCCCN(C(C2(C)C=CCC2)=O)C1 70575,N(C1CCCn2nccc21)C(C1(C=C)CCN(C(c2n[nH]c(C)c2O)=O)C1)=O 70576,Cc1ccc(C(C)CC(=O)NC(C)C(C)(C)NC(c2ccsn2)=O)cc1 70577,c1(N(C)C)ccc(-c2nc(C(=O)Nc3ccc(O)cn3)cs2)cc1F 70578,c1(OC)ccc(CO)cc1C(=O)NC(CNC(=O)CN1CCCCC1=O)C1CC1 70579,c1(C(=O)NCC(CN(C(=O)C=C2CCSCC2)C)(C)C)ccc2ccsc2c1 70580,CCC(CC(=O)NC(C(=O)N(C1CCSC1)C)C(C)O)C(F)F 70581,C12(C(=O)NCC(C)(C)C#N)CC(CN(C(C3C4CCC(F)C34)=O)C1)C2 70582,C1(C)(C(N2CCC(O)(C(C)NC(C(C)NC(N)=O)=O)CC2)=O)CCCCCCC1 70583,N1(C(c2c(CC)cco2)=O)CCCN(CCNC(=O)Cn2cncn2)CC1 70584,Cc1c(C(=O)NCC2CC(NC(C34CC(C)(C3)C4)=O)C2(C)C)cccc1O 70585,C#CC(C)(C)C(=O)NCc1nc(C(=O)NC(C)CC(C)CC)c(C)o1 70586,C(=O)(CCCCC#N)N1CC(CNC(C2(C)C=CCC2)=O)OCC1 70587,C#CC1(NC(=O)C(C)(C)CN(C)C(c2ccc(=N)[nH]c2)=O)CCOC1 70588,N1(C(=O)COC2CCOC2)CCCC(C2CCCN(C(c3ccc[n+]([O-])c3)=O)C2)C1 70589,C1(NC(CN(C)S(N)=O)=O)CCCC12CN(C(=O)CCn1cc[nH]c(=O)c1=O)C2 70590,c1(C(c2nnnn2C)NC(c2c(F)cccc2F)C)cc(F)c(Br)c(F)c1 70591,C(=O)(C(C)CC(C)C(C)=O)NCCn1cc(C(N2C(C)(CCC)CC2)=O)nn1 70592,C1(CC(=O)NC2C(CNC(C(COCC)(C)C)=O)CCCC2)CC2CCC1CC2 70593,c1(C(N(C(CNC(c2cc(C)cc(C)n2)=O)C2CC2)C)=O)ccc2[nH]ccc2n1 70594,N1(C(C(COC)(C)C)=O)CCC2(CC1)OCCCC2NC(=O)CSS(C)(=O)=O 70595,c1(C(CC)C)ccc(NC(C2CCCN2CC(=O)NCc2nccn2C)=O)cc1 70596,C#CCC(C)C(=O)N1CCC(CNC(c2ccc(C3(C)CC3(F)F)cc2)=O)CC1 70597,c1(C(C(C)C)NC(CCc2cn(CC)nc2C)=O)ccc2ncccc2c1 70598,N1(CC(C2CCCCC2)CC#C)CCC(CO)(CNC(=O)C(O)C=CC)CC1 70599,C12CCC(C1)NC2=O.c1(C(=O)NCCNC(C2(Br)CC2)=O)ccco1 70600,c1(C(N(C)CC2CN(C(c3ccn(C)n3)=O)CCO2)=O)ccc(C2CC2)c(Cl)c1 70601,C(C)(C)(C=CC(=O)NC1(CC(=O)NCC(C)SC)CCC1)SC 70602,C(CCC(C)CCC)c1nc(-c2ccc(OCC)cn2)on1 70603,c1(CC)nn(C)c(CC(N2CCCC(NC(=O)C(C)CC3CCC3)C2)=O)c1Cl 70604,C1(C(N2C(CNC(c3n(C)cc(C#N)c3)=O)CC(F)C2)=O)CNC(=O)C(C)(C)C1 70605,C(C(=O)N1CC(C(N2CCC(CC(C)C)CC2)=O)C(F)C1)(C(C)C)SCC 70606,c1(-c2nc(C(C)SC)nn2C(c2cncc(F)c2)C)cc2c(OC)cccc2[nH]1 70607,C1(NC(c2c(C)ocn2)=O)CN(C(=O)C(C)OCC(C)C)CCC1F 70608,C(CCCCC(=O)NCC(C)(C)OCCNC(C1CCC(N(C)C)C1)=O)SC 70609,Cc1nn(C(C)(C)C)cc1C(N1CCN(C(=O)COCCN(C)C)CC1)=O 70610,CC(C)C(C(=O)N1CC(C(N)=O)(CNC(C2CC3C=CC2O3)=O)C1)NC=O 70611,C#CC1(NC(C2(CNC(=O)C(C)OCCN(C)C)CC2)=O)CCOC1 70612,CCCCC(CNC(c1ccc(F)s1)=O)NC(=O)C(O)C1CCC1 70613,N1(C(CC2C(=O)OCC2)=O)CCC12CN(C(C1CCCCCC1)=O)C2 70614,Cc1c(C(=O)NCC2COC(C)(C)CN2C(=O)C=CC2CCC2)nc2sccn12 70615,c1(CCCNC(CN(CCOC)C(C2C=CCS2)=O)=O)nc[nH]n1 70616,n1(CC)nc(C(N2CC(N(C)C(c3cc(-c4ccccc4)[nH]n3)=O)C2)=O)cc1C 70617,CC(C)C(C)(O)C(=O)NC1CC1NC(c1cc(Cl)ncc1O)=O 70618,C1(N(C(=O)C(C)N(CC)CC2CC2)CCC)CCN(C(=O)Cc2cn[nH]c2)CC1 70619,c1(CN2CC(NC(C3C(C)CC(C)O3)=O)(CO)C2)ccc(S(=O)(=O)C(F)F)cc1 70620,N1(CCC)CC(C(N2CCCC(N(C(=O)Cc3ccoc3)CCO)C2)=O)CC1=O 70621,CCC(CC(=O)NCC(C1CC1)N(C(=O)Cc1cnnn1C)C)SC 70622,CC(C)CC(C)C(=O)N(C1CN(C(=O)CC2COCC2(C)C)C1)C 70623,C1(NC(c2cn(C)nc2O)=O)CC(NC(=O)CC2(c3ccon3)CC2)C12CCC2 70624,Cc1cc(C)c(C(N2CCN(C(=O)CC3COCCN3C)C(CO)C2)=O)c(C)c1 70625,c1(C(N2CCCC(OC3CC3)C2)C(=O)NCCOC)nc(Br)ccc1OC 70626,C(=O)(CC(P(C)(C)=O)P(C)(C)=O)N(C(CNC(C(CCC)O)=O)C)C 70627,c1(C(N2C(C)CCC(CNC(=O)CCC(C)(C)C)C2)=O)ccc2n[nH]cc2c1 70628,c1(C(=O)NCC(CC)NC2CN(C(c3ccn(CC)n3)=O)C2)ccc(C(N)=O)o1 70629,C(CC)(CCC(=O)Nc1ccc(OCF)cc1)NC(C(CC)CC)=O 70630,C12(NC(c3cc4n(n3)CC(F)C4)=O)CCCC1CN(C(c1cc(O)cs1)=O)C2 70631,C=CCC(F)(F)C(=O)NCC(F)CNC(c1ccc([N+](=O)[O-])o1)=O 70632,c1(C(=O)NC2CCN(C(c3ccc(OC)s3)=O)CC2F)ccc2nc(O)sc2c1 70633,N(C1CCCc2cc(CNC(=O)CCCCC3CC3)ccc21)C(C1CN(C)C1)=O 70634,c1(CNC(C(=O)NCC)=O)cccc(CNC(C2CCC(F)C2)=O)c1 70635,N1(C(C=Cc2cn(C)nc2)=O)CC2COCCC2(NC(=O)C(F)=C2CCCC2)C1 70636,C1(CNC(C2(CC#C)CCC2)=O)CCN(C(=O)CN2CCCCC2C)CC1 70637,c1(C(=O)NCC2CN(C(C(C)=C3CC3)=O)C2)ccc(C(F)F)nc1 70638,CCCC(O)C(=O)N1CCC(OCCNC(c2coc(C#N)c2)=O)C1 70639,c1(C(=O)NCC(CC(=O)NCC(CC=C)(C)C)C)cc(F)cnc1O 70640,c1(CNC2CCN(c3c(C(=O)O)ccs3)C2=O)noc2cc(Br)ccc12 70641,C(C(C)N=c1nc(OC)cc(OC)[nH]1)NC(CCC(=O)NC)=O 70642,CC(C)C(C(=O)N1CC(NC(=O)CSC(F)(F)F)C(C)C1)NS(=O)(=O)C1CC1 70643,CC1CN(C(C2CC(C)(C)CO2)=O)CC1C(=O)NC1C=CCC1 70644,C1(NC(c2ccn(CC)c2C)=O)CN(C(C23CCCC2C3)=O)C2(CCCCC2)C1 70645,C(CC(C(=O)NCC1CCCCO1)NC(=O)CC1CCC(=O)C1C)OC 70646,C(CCCCCNC(=O)CC1CCCC1)NC(c1cc(CCC)[nH]n1)=O 70647,C=C=C(C)CC(=O)NC(C1CCCN1C(=O)CCSc1nccn1C)C 70648,C(=O)(C1=CCCCO1)N(C1CCCN(C(C2(CC=C)CCOC2)=O)C1)CC 70649,N1(C(CCCOCCOCC)=O)CCN(C(=O)CN2CSCCSC2)C2CCC12 70650,C1(CC=C)(NC(C2CCN2C(C)(C)C)=O)CN(C(=O)Cc2ccsc2)C1 70651,c1(OC)ccc(C(C)NC(=O)NC(C)C(c2ccc(F)cc2)O)cc1C 70652,N#CC1CN(C(=O)C2=CCN(C(c3ccn(C4CC4)n3)=O)C2)CC12CCC2 70653,C1(NC(C2CC(NC(c3ccoc3)=O)C2)=O)CCCC(O)CC1 70654,CC(C)(CCCO)CN=c1[nH]c(=NCC2CCOC(C)(C)C2)c2sccc2[nH]1 70655,c1(C(=O)NCCCNC(CC(COC)(C)O)=O)[nH]c2ccccc2c1Cl 70656,CCCC(C(=O)NC(C)CC1CN(C(c2coc(C#N)c2)=O)C1)S(N)(=O)=O 70657,c1(CN(C(=O)NC2CCC(C)(CC)CC2)CC)cc(Br)ccc1C 70658,c1(OC)cc(C)cnc1C(=O)NC(C(C)NC(c1cn(C2CC2)cn1)=O)C(C)C 70659,C(N=c1[nH]c2c(c(=NCCCC3(C)N=N3)[nH]1)CCCC2)C1(CC(C)C)CCCC1 70660,Cn1cnc2ccc(C(=O)NCC3CC4CCC3N4C(c3cc(Cl)on3)=O)nc12 70661,Cn1ncc2nc[nH]c(=NC3CCCC(C(=O)NCCc4ccc(O)cc4)C3)c12 70662,CP(C)(=O)c1ccc(C(=O)NCC(C2CCC2)NC(c2ncccc2F)=O)cc1 70663,CC(C)(CNC(C1CC2CC1CC2O)=O)CC(=O)NCCC1(CO)CC1 70664,N1(C(C=CCNC(=O)CCC2OCCO2)=O)CC(O)CC12CCC2 70665,N1(C(CC2CN(C)CC2O)=O)CC(NC(c2ccoc2Cl)=O)C(C)(C)C1 70666,C(=O)(CC(C(=O)NC1CCCCC1NC(=O)Cn1ncn(C)c1=O)N(C)C)OC 70667,C1(C(N2C3(C(N4CCC(O)(C(C)C)C4)=O)CC3CC2)=O)C2CCC(C2)C1C 70668,c1(C(=O)NC2CC(CCC(=O)NC3(CCCC)CC3)C2)cnc(C)n1C 70669,Cc1c[nH]c(C(=O)NCC2CCCN(C(=O)CCc3nccn3C(F)F)C2)c1C 70670,N1(C(C(=O)NC2C(NC(CCCC)=O)COC2)CC)C(=O)CCC1=O 70671,N1(C(C(C)N(C(C2CC(=O)CC(=O)C2)=O)CC)=O)CC(C)CCCC1C 70672,C=CCC(CNC(=O)C(C)(C)N(S(C)(=O)=O)C)NC(=O)C(C)(C)C1CC1 70673,C(C(C)C(=O)NCCN(C)CCOC)N(C(C(C)SC)=O)C 70674,c1(C(N(C2C(C)CCN(C(CCCC#CC)=O)C2)C)=O)cc(F)cc(Br)c1F 70675,C1(C(N(CCN(CC)CC)Cc2ccsc2)=O)CC2(C1)CC(F)(F)C2 70676,c1(C2(CC(=O)NCC(CNC(C3C(OCC)C3)=O)(C)OC)CC2)ccccc1F 70677,C(=O)(C(CNC(=O)CC1CC=CCC1)C(C)(C)C)N(C1CCCCC1)CCC 70678,C1(NC(=O)CCC2CCOC2)CC(O)(CNC(c2ccc(CO)s2)=O)C1 70679,N1(C(CC2CC(OC)C2)=O)CCC2CN(C(=O)C=CI)C2C1 70680,N1(CC(=O)NCC(CO)NC(COCCOC)=O)CCS(=O)(=O)CC1 70681,N1(C(c2c(CC)ncs2)=O)CCC(C2CC2NC(C2CC(C(C)C)C2)=O)CC1 70682,Cc1cccc(C(C(C)C)NC(=O)C(=O)NCC2CC=CCC2)c1 70683,c1(OC)cc(C)c(NC(CCC(F)F)C(N)=O)cc1Oc1ccnc(CO)n1 70684,N1(C(CN(C2CCC2)C(C)=O)=O)CC2CCC(N(C)C)C2C1 70685,C(=O)(C1=CCCSC1)NCC1C(CNC(C(CCOC)C)=O)C1 70686,CCC(CC(=O)NCCCCn1cc(CC(C)(O)c2cccs2)nn1)CC(F)(F)F 70687,S(=O)(=O)(CC(=O)NC1C2CC1N(C(c1ncccc1C(N)=O)=O)C2)N(CC)CC 70688,N1(C(c2cc(C(=O)OCC)ncc2)=O)CC2CCC1CN2C(C1CC(F)(F)C1)=O 70689,C1(C(N2CC(C(N(C(CO)C3CC3)C)=O)OCC2)=O)CC(=O)NC1(C)C 70690,C(=O)(C(C)S(N)(=O)=O)N1C(CNC(c2c(C)[nH][nH]c2=N)=O)CC1 70691,c1(C(=O)NC(C2CCN(C(C=CSC)=O)C2)C)cccnc1C 70692,c1(C(=O)NC2CCC(CNC(C(C)c3ccco3)=O)CC2)ccn2cnnc2c1 70693,C1(C(=O)NC2CON(CC)C2=O)CC(C)(C)CCN1C(C1CCN1C)=O 70694,C1(C(=O)OC)CN(C(C(=O)NCc2ccccc2)C2CC2Cl)C2(CCC2)C1 70695,c1(C(=O)NCC2(F)CC(CNC(C(C)(C)N(C)C)=O)C2)cc(Cl)c(F)cc1F 70696,c1(C(=O)NCC2C(NC(C3(C)CC4CC4C3)=O)CCCC2)ccc2c[nH]nc2c1 70697,N1(C(C(C)CC2CC2)=O)CC2(C)CC1(C(=O)NCCC1(C)CCOC1)C2 70698,C(C(CC1CC1)C(=O)N1CCC1(C)CC1CCC1)NC(C1CC(N(C)C)C1)=O 70699,C=CCC(C)C(=O)NCCCC1(NC(=O)C2=CCOC2)CC1 70700,CC(C)(CCC(=O)N1CC(C(=O)NCC(c2cnc[nH]2)O)C(F)C1)[N+](=O)[O-] 70701,c1(NC(C(CC=C)CNC(C2CC3CCC(C2)O3)=O)=O)cnc(C)c(C)c1C 70702,c1(CC)ccccc1CC(N1CC(C)(NC(C2CC(C)CO2)=O)C1)=O 70703,C=CC(C)C(=O)NCc1c[nH]nc1C(N1CCCCC1)=O 70704,c1(C(=O)NC2(C)CCN(C(=O)CCc3cnoc3)C2)nccc2ccsc12 70705,C1(C(N2CCN(CCNC(=O)C(C3CC(F)(F)C3)O)CC2)=O)CC(=O)C12CCC2 70706,C12(C(=O)N(CC(N3CC4C(CO)C4C3)=O)CCO)CCCC1C2(F)F 70707,N1(C(=O)CCc2cccc(Cl)c2)CC2CC(CNC(C34CC3C4)=O)C2C1 70708,c1(SCC(=O)N(CCC(C)NC(C(CCSC)O)=O)C)ncnc2[nH]cnc12 70709,CCC(O)C(C)(C)C(=O)N1CCOC(CC(=O)NC2(C)CCCC2)C1 70710,c1(OC)ccc2c(c1F)CCC2NC(c1cncc(Br)c1)C 70711,c1(C(=O)NCC2CCN(C(CC=C)=O)C23CCC3)ccc2nc(N(C)C)sc2c1 70712,C1(CNC(CC2(C=C)CCC2)=O)CCN(C(c2ccc(N)c(O)c2)=O)C12CCC2 70713,CC1CN(C(c2cc(Br)n(C)c2)=O)CC1NC(C1CC12CC(O)C2)=O 70714,C1(C)(C(=O)NC(c2cnc(C)s2)C)C=CCN1C(c1cnn(C)c1Cl)=O 70715,C(=O)(C(F)(F)C1=CCOCC1)N(c1cc(N)c(Cl)c(O)c1)C(=O)OC(C)(C)C 70716,c1(C(N(CC(C)O)CCNC(C(C)OCC)=O)=O)cnc(CC(C)(C)C)o1 70717,C(c1ccc(F)cc1)=CC(=O)NCC1(C(=O)Nc2ccc(F)c(F)c2)CC1 70718,C(C(CO)(CO)NC(=O)CC1(C)CCC(=O)N1)N(C(=O)C=Cc1cn(C)cn1)C 70719,CC(C#N)C(=O)NC(Cn1cccn1)C(=O)N(C)Cc1ccsc1 70720,C(=O)(CC(C)CC(C)C)NCC1(CC)CN(C(C2CN(C)CCO2)=O)C1 70721,n1(CC(=O)NCC(Cc2cccnc2)C(=O)O)cc2ncccc2n1 70722,c1(C(=O)NCCN(CCC)C(C2CNC(=O)C2)=O)ccc(COC)cc1 70723,C1(CC(C)NN(C)Cc2ncoc2C(F)F)Cc2ccccc2O1 70724,CC1C(NC(C2CCCO2)=O)CCN1C(=O)Cn1ccnn1 70725,C1(CC(N2C(CNC(c3c[nH]c(=N)o3)=O)CC2)=O)CC(C2CC2)C1 70726,c1(NC(c2ccc(C=C)cc2)c2nnnn2CC)ccc2nc(Cl)cc(C)c2c1 70727,c1(C(=O)NCC2N(C(CC3CCC(=O)C3)=O)CC(F)(F)C2)nc2c(s1)CCCC2 70728,N1(C2C(NC(C3CCOCC3)=O)CCC2)CCN(C(C23CCCC2C3)=O)CC1 70729,CC(C(=O)NCC1(CNC(=O)CCn2cncn2)CC12CCC2)S(C)(=O)=O 70730,c1(C(=O)NC2(C)CC(NC(C(C)Cc3cnc[nH]3)=O)C2)cnc2c[nH]nc2c1 70731,Cn1nc(C(=O)NC2CN(C(=O)CC3CCOCC3)C3CC23)c2ccccc12 70732,c1(C(=O)NCC2N(C(C(CC)NC(C)=O)=O)CCCCC2)cccc2sncc12 70733,O=C(CC1=CCCCC1)NC1CCCN(C(=O)Cn2ccnn2)CCC1 70734,C1(CS(C)(=O)=O)CN(C(C2CCCCCCC2)=O)CCN1C(C12CC(F)(C1)C2)=O 70735,C(=O)(CC(C)(C(F)(F)F)N(C)C)N1CCC(N(C(=O)C=CCCC)CC#C)CC1 70736,C1(C)(NC(=O)NCCCC(=O)N(C(CF)CF)C)C=CCCC1 70737,C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NCC(C)(C)NC(C(N1C(C)CCC1C)=O)=O 70738,N1(C(c2ccn(C)n2)=O)CCC2OCCN(C(=O)C(O)C(F)F)C2C1 70739,C=C(Cl)C(C)(C)C(=O)NCC12CCC(CC1)N2C(c1sc(COC)nc1C)=O 70740,Fc1cncc(C(c2nc(-c3cccc(Cl)c3)nn2Cc2ccccn2)OC)c1 70741,c1(CNC(C(=O)NCC(n2cccn2)C)=O)ccc(CN2CCNC(=O)C2)cc1 70742,CC(CC(=O)NCC(CC(=O)N1CC(N2CCNC2=O)C1)C1CCC1)C(F)F 70743,C(=O)(C(C(C)C)C(C)C)NC1C(NC(c2c(Cl)c(C)n(C)n2)=O)CCCC1 70744,Cc1nsc(C(=O)NC2CC(CNC(=O)C(O)C3CCC3)C2)c1N 70745,N1(C(CC2CN(C)C2)=O)CC(NC(=O)COC2CCCC2(C)C)C2(CCC2)C1 70746,C12CC(C(F)(F)F)CN1C2=O.C1(CN(C23CC(F)(C2)C3)C(C)=O)CC(C)(C)CO1 70747,C1(CNC(C2(N(C)C)CCCC2)=O)CCC(NC(=O)Cc2cnccn2)CC1 70748,c1(CC)c(C(=O)NC2(CF)CCN(C(C3CCC(CN(C)C)O3)=O)C2)cnn1C 70749,CC1(C)C2CCC(C(=O)NCC3(O)CCN(C(=O)CNC=O)C3)C1C2 70750,C1(CNC(C2C(CC)CCO2)=O)COC(C)(C)CN1C(c1cc(N)ccc1C)=O 70751,c1(CC)cnc(C(=O)NC2(CN3CCN(C(C4CCC(F)C4)=O)CC3)CC2)cn1 70752,c1(N(CCC(C)O)C)nc(=NC(C)CC(N)=O)[nH]c2ccccc12 70753,N1(C(C(C)SC)=O)CC(CNC(=O)Cc2cccc(NC(C)=O)c2)C(C)C1 70754,c1(C(=O)NCCOC2CCN(C(CC3C(C)C3)=O)C2)cc(C#N)ccc1F 70755,C1(CC(N2C(CO)CC2C)=O)(OC)CN(C(=O)C=Cc2ccoc2)C1 70756,c1(N2CC(CNC(=O)Cn3nnnc3C3CC3)OCC2)ncnc2[nH]cnc12 70757,C1(c2n(C(C)C3CC3)nnn2)(NC2(CO)CCOC2)CC2(C1)CC(C)(C#N)C2 70758,C1(CC)C(NC(=O)CCOC(C)CC(C)C)CCN1C(C1(c2cccs2)CC1)=O 70759,CC1(C(=O)NC(C)(CNC(c2ncccc2C2CC2)=O)C2CC2)CCOCC1 70760,c1(C(N(C2CN(C(CCC=C)=O)C2)C)=O)cccc(OC)n1 70761,C#Cc1ccc(NC(=O)C#CC(C)(C)CNC(c2cncnc2C)=O)c(C)c1 70762,C(=O)(CCCC(=O)NC1CCOC(c2ccccn2)C1)N(CC)CC 70763,CN1CCC(C(=O)NC(C(=O)NCC2(C(C)(C)O)CC2)C2CCC2)C1=O 70764,c1(CN(C(=O)CCN2CCC(F)C2)C)ccccc1CNC(=O)CC(F)(F)F 70765,c1(CC)ccccc1CC(=O)NCC(C(C)C)NC(C1CCCC1F)=O 70766,N1(C(COCCCCC)=O)CCC(C(=O)Nc2cccnc2C)CC1C 70767,C1(C)(CNC(C(CC)CCOC)=O)CN(C(C23CC(C)(C2)C3)=O)C(C)(C)C1 70768,N1(C(c2c(C)csc2)=O)CCC(n2cc(-c3cscn3)nn2)C(O)C1 70769,N1(C(c2cc(CC)n(C)n2)=O)CC(NC(=O)Cc2nccn2C)C(C)(C)C1 70770,N1(C(=O)OC(C)(C)C)CC2(CCN2C(=O)CCC(c2ccc(C(N)=O)cc2)=O)C1 70771,c1(C(=O)NCC(N2CCCC(C(=O)OC)C2)=O)cc(S(C)(=O)=O)cc(F)c1Cl 70772,CC1(C)CC(NC(=O)C(=O)NCC(F)(F)F)CN(C(=O)C(C)(C)S(C)(=O)=O)C1 70773,c1(C(=O)NCCOCCN(C(=O)C(C2CC2)C2CC2)C)ccc(Cl)s1 70774,C(=O)(CC(C)CNC(C1COCC(C)O1)=O)NCCc1cnc(C)[nH]1 70775,C1(NC(=O)COC2CCOC2)CCC(CNC(=O)COc2ccc(Cl)nc2)CC1 70776,C1(C2CN(C(=O)CNc3ccccn3)C2)CN(C(c2ccc(CO)s2)=O)CCO1 70777,O=C1Cc2ccc(C(N3CC(CNC(=O)CCCN=[N+]=[N-])C4CC34)=O)cc2N1 70778,N(C1CCc2cccnc21)C(c1cc(-c2c(C3CC3)cccc2F)ccn1)=O 70779,c1(C(N2CCC3C(NC(C4(F)CCCCCC4)=O)C3C2)=O)ccn2cncc2c1 70780,S(=O)(=O)(c1ccc(N(C)CCc2ccc(Cl)cc2)cc1Cl)NC(C)CCCO 70781,C1(C(=O)NC2(CF)CN(C(c3c(C)nc(C4CC4)o3)=O)C2)CC2CCC(C1)C2 70782,c1(C(=O)NCC2(F)CN(C(C3C(CC)CCC3)=O)C2)cc(Br)cnc1S 70783,c1(CCC(=O)NCC(C2CC2)NC(=O)C(F)c2ccsc2)nc(C2CC2)no1 70784,C1(CCN(C(=O)Cc2cccnc2Cl)C)CCCCN1C(=O)CC1CCC1(C)C 70785,C(=O)(C(O)C(F)(F)F)NC(C(C)O)C(=O)NCCOCCN(C)C 70786,CCCC(C)CC(=O)NC(CNC(c1cc(C)cnc1Cl)=O)CC(C)C 70787,C1(NC(c2c(C#C)c[nH]n2)=O)CCCCCCC1NC(=O)CCCCOC 70788,N#Cc1ccccc1C(N1CC2CCC2(CCNC(=O)C=Cc2ccsc2)C1)=O 70789,c1(CCC(=O)N(C2CCN(C(=O)C=NOC)C2)CCC)cn(C)nn1 70790,C1(C2CC2)(C(=O)NC(CC(=O)NC)C2CC2)CN(C(C2CC(SC)C2)=O)C1 70791,C(=O)(CC(C)(O)C(F)(F)F)N1C(CNC(C2CCS(=O)(=O)CC2)=O)CC(C)(C)C1 70792,c1(C(N2CCOC(CNC(c3cc(CO)[nH]n3)=O)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 70793,C1(C(=O)NC2(CCNC(CN3CC(CC)C3)=O)CC2)CCN(C(C)=O)CC1 70794,c1(CNC2CC(CN=[N+]=[N-])C2)cc(O)c2ccccc2c1 70795,C1(C(=O)NCC(CC(C)C)NC(=O)C(C)(O)C(C)C)CCCCNC1=O 70796,c1(C(N2CCC(CNC(C(C(CC)C)C)=O)C23CC3)=O)cnc2c(c1)ncn2C 70797,Cc1cccc2cc(C(=O)N(CC(C)(C)NC(c3occc3Br)=O)C)cnc12 70798,C=CC1(C(=O)N(CCCN(C(=O)C(C)Cc2ccncc2)C)C)CCC1 70799,c1(C(C(=O)NC2CC2)N(C)CC2CCCC2O)ccc2ccc(Br)cc2n1 70800,O=C(C1=CCCCO1)NCCCOCCNC(C1COC2(CO)CC1C2)=O 70801,C1(C(=O)NC2CCOCC2C)(CC)CCN(C(c2csnn2)=O)C1 70802,CC1(C)CC(C(=O)NCC2CN(C(=O)C3CC3)CC23CC3)CCO1 70803,O(NC(=O)C(O)C1CN(C(C2COC(=O)N2)=O)C1)CCCCCN(C)C 70804,C#CCCC1=C(C(=O)OC)C(c2nc(C)[nH]c2Br)NC(=S)N1CC1CC1 70805,C1(NC(C=C(NC(C)=O)C)=O)CC2CCC(C1)N2C(=O)Cc1ccccc1O 70806,C(=O)(C(CO)C(C)(C)C)N1C(C(N2CCN(CCOC)CC2)=O)C2CCC1C2 70807,c1(C(N(C(C)C)CCNC(=O)CCCCc2cnn[nH]2)=O)ccnc2[nH]ncc12 70808,C1(NC(C2C(C)(Br)C2)=O)CCC2CN(C(C3(C#N)CCCCC3)=O)CC2C1 70809,c1(C(N(CCNC(C2CN3CCN2CC3)=O)CC)=O)ccc2c(c1)N(C)CCO2 70810,N1(C(C(C)C#N)=O)C2CCC1CC(CNC(c1cc(Cl)ccc1OC(F)F)=O)C2 70811,C1(CCNC(C2CC(OC)C2)=O)CN(C(C2CCN2C2CCCC2)=O)CCO1 70812,c1(OCC)cc(F)ccc1C(N1CC2C(C1)N2C(c1cnco1)=O)=O 70813,C12(NC(c3n(CC)ncc3)=O)CCC(C(N3CCC(C)(O)C3)=O)(CC1)CC2 70814,CCCC(CCCNC(=O)COc1ccc(F)cc1)NC(C1(C)CC1C)=O 70815,c1(SCC)ccc(Cl)cc1NC(c1c(OCCC)cccc1F)=O 70816,c1(C(=O)NCCOCCN(C(C(CC#C)C)=O)C)cc2c(nn1)CCCO2 70817,Cc1cc(C(=O)NC2CCCCC2NC(C2CCC(=O)O2)=O)cc(C)c1Br 70818,Cn1cc(Br)c(C(=O)NCC2(CCNC(=O)Cn3cccn3)CC2)cc1=O 70819,Cc1cc([N+](=O)[O-])c(N2CCC(C(F)(F)F)C2)cc1Br 70820,C#CC1CC2(CC2)CN1C(=O)C(C(C)CC)N(C)C(c1oc(C)cc1C)=O 70821,c1(CNC(c2ccccc2Cl)c2n(CC)nnn2)ccc(Cl)nc1 70822,c1(NC(C(=O)NCC(=C)F)=O)cc(C(F)(F)F)ccc1OC 70823,c1(NC(c2noc(C3CC3)n2)CC)cc(C(=O)C(F)(F)F)ccc1F 70824,C(=O)(C(O)CC(F)(F)F)NC1(CC(N2CCC(C(=O)OC)CC2)=O)CCC1 70825,N1(C(CC=C=C)=O)CCCN(C(c2ccc(OC)cc2C)=O)CC1 70826,C1(C(=O)NCC(CCOC)OC)(CNC(C2CCC(CO)CC2)=O)CCC(O)CC1 70827,C1(C(N(C2CCCC2)CCCNC(C(c2cncnc2)C)=O)=O)CCC(C)(C)O1 70828,C1(NC(c2cn(CC)nc2)=O)CCC(NC(=O)C(C)Sc2ccc(F)cc2)CC1 70829,N1(C(C(C)OC2CCOC2)=O)CCC(NC(=O)CCCN(C)C)C(O)C1 70830,N1(C(C2(C(C)C)CCN(C(c3ccsn3)=O)C2)=O)CCC12CCSCC2 70831,C(CCCCC(=O)N1CCCC(C(C)(O)CNC(c2cc[n+]([O-])cc2)=O)C1)OC 70832,C1(C(=O)NC(C)CCNC(c2occc2F)=O)C2CCCOC12 70833,N1(CC)Cc2ccc(NC(=O)NC3CCc4ccccc4C3)cc2C1 70834,C1(N(C(C(=O)OC)C)C)CCSCC1.c12noc(n1)C2SC1CCCCC1 70835,Cc1ccc(CCC(N2CCN(C(c3nnc(O)nc3O)=O)CC2)=O)cc1Cl 70836,CN1CC(=O)N(CC(=O)NC2CC(NC(=O)Cc3cn(C)cn3)C2)C1=O 70837,C1(C(N2C(CNC(c3cc(CC)on3)=O)CC2)=O)CCOCC12CCC2 70838,Cc1[nH]c(=NC(=O)N2CCc3[nH][nH]c(=N)c3C2)ccc1C#N 70839,N1(C(c2nccc(C)c2)=O)CC2CCC1C(CNC(c1cccc(O)c1C)=O)C2 70840,c1(CN2CCN(C(C3CC(OC)C3)=O)C(C)C2)nc(C)nc2sc(C)c(C)c12 70841,c1(C(C(=O)NCC2N(C(c3nccc(COC)c3)=O)CC2)O)cc(Cl)cc(Cl)c1 70842,N1(C(C(=O)NC(c2ccc(Nc3ccccc3)cc2)=O)=O)CC2CCNCC12 70843,C1(CC(=O)NC(CC)(C)CO)CN(C(c2c[nH]c(=N)o2)=O)CCO1 70844,C(=O)(CC1=CCCCC1)NCCC1(C)CCN(C(CC)C(=O)NCC(C)OC)C1 70845,Cc1cc(C(=O)NCC2CC(NC(=O)C=CC(C)(C)C)C2)n(C(C)(C)C)n1 70846,c12cccc(c1)NC2=O.C1(NC(C2CC2C)=O)CCCC1N.CCS(=O)(=O)NC 70847,C(=O)(C(C(C)(C)C)NC(C1(Cl)CC1(F)F)=O)NCCC(C)N1CCCC1 70848,c1(-c2cn(C3C(C)CN(C(=O)C(F)C4CCC4)C3)nn2)cc(Cl)cc(Cl)c1Br 70849,C1(CC)C(=O)CC1C(=O)NC(c1ncco1)(C)C 70850,C=Cc1cnn(C)c1C(=O)NC(C1CCN(C(=O)C(C2CCCCC2)F)CC1)C 70851,c1(OC(F)F)cccc(NC(c2nnnn2C(c2ccco2)C)C2CC2(C)C)c1 70852,C1(NC(c2ccc(CCC)cc2)=O)CCN(C(c2cnc(N)c(O)c2)=O)CC1F 70853,C(C1=CCSC1)(c1n(C(C)CCc2ccccc2)nnn1)NCC(CO)C(C)C 70854,C1(N(C)C(C2CCN(c3ncccn3)C2)=O)CC1C1CC1 70855,C1(NC(C2(CC)CN(C(C(CCCC)C)=O)C2)=O)CCCCC12CCC2 70856,C1(CNC(c2scnc2Cl)=O)CN(C(c2cn[nH]c2)=O)C2(CCOCC2)C1 70857,N1(C(C(C)(C)NC(=O)OC)=O)CCN(C(=O)C(C)c2cccs2)C(CN(C)C)C1 70858,c1(CC(=O)NC(CC#C)COC)nc(C)ccc1Br 70859,c1(C(N2CCC(NC(c3c(OC)scc3)=O)CC2C)=O)cc(C)cc2ccoc12 70860,c1(C(=O)NCCC(CNC(C2(CCC)CCC2)=O)O)cc(Cl)c2[nH]c(O)nc2c1 70861,c1(NCC(=O)NCCCCNC(C2CCN(C(C)=O)C2)=O)cc(C)n(C2CC2)c1 70862,C1(C(=O)NC(C)CCNC(c2ccnc(Cl)c2N)=O)CC(C(C)(C)C)=NO1 70863,C(C(C)(C)C(=O)N1CCC(OCCF)C1)N(CC(=O)NC1CCC1)C 70864,C(C(=O)N1CCOC(CC(N2CC(O)CC2CN(C)C)=O)C1)(C(C)C)OCC 70865,c1(CC)cccc(OCC(=O)NCCC(C)(C)NC(C2CCC(C)O2)=O)c1 70866,c1(CC)ccc(C(N2CCC(C)=C(Br)C2)C(=O)NC2CCOCC2)cc1C 70867,C(=O)(C(C(C)C)SCC)NC1(CCNC(C2(CC#C)CCOC2)=O)CCCC1 70868,c1(C(=O)NCC2N(C(C(=O)NCC)=O)CC3(CC3)C2)cn2c(n1)CC(OC)CC2 70869,C(=O)(C(C)(C)CCCNC(=O)CCc1nccs1)NCCOCCN(C)C 70870,C(=O)(N=c1[nH]nc(CC#N)s1)N1CCC(CN(CCC)CC)C1 70871,C1(C(CNC(C(C)(C)n2ccnn2)=O)(C)O)CCN(C(C2CCCCC2)=O)CC1 70872,C(CC(CNC(=O)Cc1cn[nH]c1)OCC)NC(C(C)OCC#C)=O 70873,CN1CC(NC(c2cc(CNC(c3ccc(O)nn3)=O)ccn2)=O)CC12CCC2 70874,CCCCC(CC)NC(N1CCCC(COc2ccccc2)C1)=O 70875,C#Cc1cc(C(N2CCC(F)C(NC(=O)Cc3ccccc3)C2)=O)cc(N)c1 70876,N1(C(C2(COC)CC=CC2)=O)CCC(F)(CNC(C2(COC)C=CCC2)=O)CC1 70877,c1(OC(C)C)cccc(CC(=O)NC2CC2)c1.C1CC1NC(C1(C)CC1)=O 70878,O=C(CCC[N+](=O)[O-])N1CCOCC(CNC(C2(c3ccccn3)CC2)=O)C1 70879,CC1CCC(CCC(N2CC(O)(CNC(=O)CC34CC(C3)C4)C2)=O)O1 70880,N1(C(c2c(C(C)C)con2)=O)CCCC(C)(C(=O)NC2COCC2CO)C1 70881,CCCCC(C(=O)N(CC(C)NC(c1nn(C)nc1C(=O)OC)=O)C)C(C)C 70882,c1(C(N2C(C)CC(NC(c3ccc(F)c(F)c3)=O)C2)=O)cnn2c1N(C)CC2 70883,c1(C(=O)NCCN(CCC)C(c2c[nH]nc2CC)=O)c(C)csc1Cl 70884,C1(CNC(c2cnc(O)o2)=O)CC2(CCC2)CN1C(c1ncoc1C1CC1)=O 70885,C(=O)(CC(C)(C)C(=O)N1CC2CC(NC(c3cc(Br)cn3C)=O)CC2C1)OC 70886,N1(C(C=Cc2ccn(C)c2)=O)CC(NC(C2CC3(C2)CC3F)=O)CC(F)C1 70887,CC#CCCC(=O)NC1CCC(CCC(N2CCN(CCCO)CC2)=O)C1 70888,c1(C(N(CCN(C(=O)C(F)(F)c2cscn2)C)C)=O)ncc(C(C)(C)C)o1 70889,C1(SC)CC(NC(=O)Cn2cc(-c3csc(-c4ccc(Cl)cc4)c3)nn2)C1(C)C 70890,CCC(CC)C(F)C(=O)NCC1(CNC(=O)C(CC)OC)CCCCC1 70891,C(CC1CC1)(C(=O)NCC=CCNC(c1cc(Br)co1)=O)OC 70892,C=C(C)C(CC(=O)NC(C)(CNC(c1cc(O)ccc1O)=O)C1CC1)OCC 70893,C1(C(N2CC(CCNC(c3c(CC)con3)=O)C2)=O)CCCN(C)C1 70894,C1(C(=O)NC(C(C)C)(C)CNC(=O)CN2CCC(CO)CC2)CCCCC1(F)F 70895,C1(C(=O)NC(C(=O)NC(C(=O)NCC)CC)CCC2CC2)C2CCC(C2)C1C 70896,c1(CC(=O)NC2CC2NC(C2CC3OC(=O)CC23)=O)nc([N+](=O)[O-])n[nH]1 70897,N1(CCn2c(C)csc2=O)CCCN(C(c2c(Cl)nn(C)c2Cl)=O)CC1 70898,c1(CNC2CCN(c3cn(C)nc3)C2)cc(Br)cnc1S 70899,CC(C)CC(O)CN=c1cc[nH]cc1S(=O)(=O)N1CCc2c(C)cccc2C1 70900,c1(OCC)ccc(NC(c2nnnn2C2CC(F)(F)C2)(CC)C2CC2)c(F)c1 70901,c1(CN(C)C(C2CN(c3ccncc3)C2)=O)ccnn1C 70902,CCC(C)C(O)C(=O)NC1(CO)CN(C(=O)C(C)(O)C2CC2)C1 70903,CN1C(=O)OCC1C(N1CCC(F)(C(=O)NC2CC2)C1)=O 70904,N#Cc1cnn(CCO)c1NC(=O)NC1(c2ccc(OC(F)(F)F)cc2)CC(O)C1 70905,Cc1cnn(C(C)C(=O)NC(c2cccnc2)C(=O)NC2CC(C(N)=O)C2)c1 70906,N1(C(CC=C(C)C)=O)CCN(C(c2ccc(C(F)F)o2)=O)CC1c1cn[nH]c1 70907,C(CO)(CCCCNC(c1ccc(C2CC2)cc1)=O)NC(C=CC(C)(C)SC)=O 70908,c1(N(c2nccc(C(C)C)n2)C(C2CCCNCC2)=O)ncc2ccccc2n1 70909,Cc1cc(C(N2CCC23CN(C(=O)CCC(C)(F)F)C3)=O)c(O)c(C)c1 70910,N1(C(C)(C)C)CCCC(C(=O)NC2CN(C(C3(n4cnnn4)CC3)=O)C2)C1=O 70911,C(C(C(=O)N1CC2OC(=O)OC2CN1C)NC(C)=O)c1cc(C(=O)OC)c(C)o1 70912,c1(OC)cc(C)cnc1C(=O)NCC1C2CN(C(c3nn(C)cc3Cl)=O)CC12 70913,Cc1cc(C)n(CC(N2CCC2CNC(c2cc(Cl)c(F)cc2N)=O)=O)c(=O)n1 70914,Cc1ncc(CC(=O)NC2CCC2CNC(=O)CCCN(C(C)(C)C)S(C)(=O)=O)s1 70915,c1(C(=O)NCC2CCC(C(NOC(C=C)C)=O)C2)cnc[nH]c1=N 70916,CCC(C(=O)NC1CC(C)N(C(=O)Cc2cc(C)n(C)n2)C1)C(C)(C)CC 70917,c1(C(=O)O)ccnc(N2CCCC2)n1.C12CCCC1C(=O)N(C(=O)CCCF)C2 70918,c1(N2CC(C(N)=O)OCC2)nc2cccc(F)c2c(=NCc2cnc(O)[nH]2)[nH]1 70919,C1(CNC(C(C#C)(C)C)=O)CN(C(=O)Cc2cc(C)on2)CCCO1 70920,Cc1cc(Br)cc(C)c1C(=O)OCC(=O)NCC(c1ccccc1)C 70921,N=c1nc(O)c(CC(N2CCCC(C)(NC(C3CC(=C4CCC4)C3)=O)C2)=O)c[nH]1 70922,c1(CN(C(COCCNC(c2ccc(CC)[nH]2)=O)=O)C)ccc(C)cc1 70923,c1(COC)ccccc1NC(C1CC1C(=O)Nc1cc(CS(C)(=O)=O)on1)=O 70924,c1(C(N2C(C)CC(NC(c3cnc(CCCC)s3)=O)C2)=O)cc2ccccc2o1 70925,O=C(C(F)(F)CO)N1CCC(OC2CN(C(=O)Cn3ccc(C4CC4)n3)C2)CC1 70926,CCCC(C)(C)C(=O)NCC1(CNC(=O)Cc2ccc(OC)cc2)CCC1 70927,c1(OCCOC)cncc(C(=O)NC2CC(CNC(=O)C(Br)=C(C)C)C2)c1 70928,C(CC(=O)N(CC(C)CO)C)(C(C)CC)NC(C(CCC)N(C)C)=O 70929,C1(CC(N2CCC(C(C)C)C2)=O)COCCN1C(=O)Cc1cc[nH]n1 70930,C(C(=O)N(C)CC1CCSC1)(C(C)(C)C)NC(c1nc(C)c(C)s1)=O 70931,c1(C(=O)NC2CN(C(CC(C(C)C)C)=O)CC2(C)C)c2c(nn1C)CCCC2 70932,c1(C(=O)NCC(CNC(c2cc(CCC)[nH]n2)=O)(C)C)ccc2oc(S)nc2c1 70933,c1(C(N2C(CNC(C(C)(C)OCC)=O)CCC2)=O)cnccc1C#N 70934,N1(C(C(C)OCC(C)C)=O)CC(C2CCCN(C(c3cc(CO)[nH]n3)=O)C2)C1 70935,c1(C(=O)NCc2cc(C(=O)NCCC(COC)O)n(C)n2)ncc(F)cc1N 70936,CC1CC(CNC(=O)C=CC2CCCCCC2)CCN1C(c1nn(C)cc1Cl)=O 70937,C1(C(N2CC(F)(C(=O)Nc3ccc(OC(C)C)cc3)C2)=O)CC(=O)OC1(C)C 70938,c1(CN(CCCC)C(c2nc[nH]n2)=O)ccccc1-c1ccc(NS(C)(=O)=O)s1 70939,CC1CN(C(=O)CCC(C)(C)NC(=O)C(C2CCCCC2)=O)CC(C)C1O 70940,C(=O)(CS(C)(=O)=O)NCC(=O)NCC(=O)NC(C)CO 70941,Cc1ccc(CNC(=O)C(CC2CC2)NC(c2cnn(C)c2)=O)s1 70942,C1(C(N2CCC(O)C(F)C2)=O)CCCCCN1C(=O)C=Cc1ccc(O)cc1 70943,C(=O)(C(O)CC(C)(C)C)NC(CNC(c1c(C)cc(OC)nc1)=O)CO 70944,c1(C(=O)NC(CCNC(CC2(OC)CCCCC2)=O)C)ncn2cc(Cl)ccc12 70945,c1(NC(c2c(N(C)C)scn2)=O)ccc(Br)c(C(F)(F)F)c1 70946,N(C)(C(=NCC1CC2CC1C2)NCC(C)(C)C)CCCOC 70947,C(CCCCCNC(C1CC(C)(O)C1)=O)N(C)C(c1nc(Cl)c(Cl)s1)=O 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70983,N1(C(CSC(C)C)=O)CCC(NC(=O)C(c2ccc(Cl)s2)C)CC1C 70984,c1(OC)cc(C(N2CCC(C)C2CNC(C2CCCCN2N=O)=O)=O)cc(C)n1 70985,c1(CCC(=O)NCCCCNC(C23CC(F)C2C3)=O)ccc(C(F)(F)F)cc1 70986,C1(N(C)C)CCC(N(C(=O)CC(O)C2CCCC2)C)CC1 70987,CC(C)C(C(=O)NCc1cncc(C(N2CC3CC2C2CC32)=O)c1)C(C)C 70988,C1(N(C(C2CCC(C)CC2)=O)C)CN(C(=O)C(C)N2CCCC2)CCC1O 70989,Cc1cc(F)c(C(=O)NCC2CCN(C(c3cnc(O)c(Cl)c3)=O)C2)c(Br)c1 70990,CC(CC(F)(F)F)C(=O)N1CCN(C(=O)COCc2nccs2)CC1CCO 70991,c1(CC)cccc(CNC(C2CCC(CNC(C3CC=CCC3C)=O)O2)=O)c1 70992,C1(CNC(CN(CCC)C)=O)C(C)CCCN1C(=O)C(C)N(CC(F)(F)F)C 70993,C1(COC(C)C)COCCN1C(=O)NC1CC2(C1)CC2NC(C)(C)C 70994,C(=O)(C(C)CC(F)(F)F)NCCOCCN(C(C(C=C)(C)O)=O)C 70995,C1(C(N2CCC(=CCNC(C3CC(=C4CC4)C3)=O)CC2)=O)CCC2(CCC2)CO1 70996,c1(C(N2C(C)(C(N(OC)CC3CC3)=O)CC(O)C2)=O)coc2c1CN(C(C)=O)C2 70997,c1(C(N2CCC3C(NC(C)=O)C3CC2)=O)cc2cccc(Cl)c2o1 70998,CCC(c1ccccc1)=CC(N1CCC(C)N(C(=O)CCC2CCCO2)CC1)=O 70999,C(=O)(C1COc2ccccc21)N1CC(CNC(C(c2cccc(Cl)c2)CC)=O)C1 71000,N1(C(c2sccc2NC(N)=O)=O)CCCC1CNC(CC1N(S(C)(=O)=O)CC1)=O 71001,c1(C(N2CCC(C(C)NC(C(C)OCC#C)=O)CC2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 71002,CC(C)CC(=O)N1CCC(CN(C(=O)CC2C(CO)C2(F)F)C)C1 71003,c1(C(=O)NC(C)C(C)C(N2CCC(C)(C#N)C2)=O)cccc2[nH]ccc12 71004,N1(C(C(=O)Nc2c(C)cc(F)cc2)C2CCCC2)CCN(C(=N)NC(=N)N)CC1 71005,CC1(C(N2CCC(OCC3CC3)C2)=O)CCCN(C(=O)CCN2CCOCC2)C1 71006,N1(C(CSCC=C)=O)CC(NC(c2cnc(CO)nc2C)=O)CC12CCCOC2 71007,C1(NC(Cc2c(C)nsc2)=O)C=CCN(C(=O)Cc2cccc(F)c2)C1 71008,C12(NC(CN(CC(=O)NC(C)C)C)=O)CCOCC1CN(C(=O)CS(C)(=O)=O)C2 71009,C1(NC(c2c(CC)cco2)=O)CCC(C)N(C(c2cnn(C)c2Br)=O)C1 71010,N1(C(=O)C(O)CCn2cncn2)CCCC(F)(CNC(C2(F)CC2)=O)C1 71011,C#CCC(CC(F)F)C(=O)N1CC(CC(=O)NC2(CC=C)CCCC2)CC1C 71012,c1(SC)cc(C)c(C(N2CC(NC(c3cc(CCO)on3)=O)C(C)C2)=O)o1 71013,C1(C(N2C(C)(CC(=O)NC(C#C)(C)C3CCC3)CC2)=O)CCCC(=O)C1 71014,CS(=O)(=O)c1ccc(CCNC(C2CC2c2cccc3ccccc23)=O)cc1 71015,N1(C(c2c(C)scc2)=O)CCCCCC1C(=O)NC(c1nn[nH]n1)C1CC1 71016,C#CC1(C(N2CCC(O)C2)=O)CCN(C(c2cncc(C#C)c2)=O)C1 71017,N1(C(C=CCOC)=O)CCOCC1CCNC(=O)C(c1ccn(C)n1)C 71018,c1(NCCOC)ncc(S(=O)(=O)N2CCC(NCC3CC(SC)C3)CC2)cc1Cl 71019,C1(NC(CSCCC(C)C)=O)CC12CCN(C(C1CCC(C)CC1)=O)C2 71020,c1(CCC(=O)NCCCN(C(=O)CC2CSCCO2)CC)nnc(C2CC2)o1 71021,c1(C(=O)Nc2ccc(C(=O)OC)c(Cl)c2)cc2ccoc2cn1.C123CC1CN(C2)C3 71022,CC1(CNC(C2CC(NC(=O)Cn3cccc3)CCO2)=O)NC(=O)NC1=O 71023,c1(C(=O)NCC23N(C(CCCC=C)=O)CCC2CCC3)ccc2c(c1)CCCO2 71024,c1(C(=O)NCCNC(=O)CSCC2CCCO2)cc(=O)n2ccccc2n1 71025,N1(C(C(C)C2CCOC2)=O)CCOC(CNC(C2(C3CC3)CCC2)=O)C1 71026,c1(CC(=O)NC2CN(C(C3(CC#C)CCCCO3)=O)CC2F)ccc(C)c(F)c1 71027,c1(OC)ccc(Cl)c(C(=O)NC2CC(F)(CNC(=O)C(F)(F)C3CC3)C2)c1N 71028,c1(NC(COC)C2CC2)nc2ccc(S(=O)(=O)N3CCSCC3(C)C)cc2s1 71029,Cc1cc(OCC(N2CC3CCOC3(CNC(=O)CC3CC3)C2)=O)cc(C)c1Cl 71030,c1(CN2CCC(O)(C(=O)NC3CC(=O)OC3)C2)c[nH]c2ncc(Br)nc12 71031,CCC(C)C(C(=O)N1CCCN(CCO)CC1)NC(c1ccc(C(C)C)o1)=O 71032,c1(NC(C(=O)N(CC(C)NC(=O)CCF)C)=O)ccc2c(c1)OCCO2 71033,CCC(C)(COC)C(=O)NC1CC(NC(=O)C(C)N(C)C)C(O)C1 71034,c1(C(=O)NC(C2(O)CN(C(=O)CCNc3ccccn3)C2)C)ccoc1Br 71035,c1(OC)cc(CNc2cccc(F)c2C(N2CC(O)C(F)C2)=O)c(Br)cc1O 71036,Cc1nn(C)c2c(NCCN3CCCOCC3)nc(=NCC(C(C)C)N(C)C)[nH]c12 71037,N1(C(N2CCC(c3nc(C)on3)C2)=O)CCC(O)CC1CO.n12nc(C)cc1C2 71038,Cc1c(C=CC(N2CCC(CCNC(C3CC4C=CC3O4)=O)CC2)=O)cnn1C 71039,Cn1cc(C(=O)NC(=O)CNC(=O)CC(O)C2CCCC2)nn1 71040,N1(C(C2(CCC=C)CCCC2)=O)CCN(C(=O)Cc2cnn(C)c2)CC1CCC 71041,c1(C(=O)NC2CC(N(C(Cn3c(C)ccc3C)=O)C)C2)ccc(P(C)(C)=O)nc1 71042,c1(C(=O)NCC(CCNC(C(C)CS(C)=O)=O)(C)C)scc2c1OCCO2 71043,CC(CNC(c1cc(O)cc(F)c1)=O)C(F)C(=O)NCC1(C(F)(F)F)CC1 71044,c1(NC(=O)NCCNS(C)(=O)=O)ccc(N2CCCC2c2cccnc2)nc1 71045,N(C(=NCc1ccn(C)c1)NCc1cccc(OCC(F)(F)F)n1)C(C)C1CC1 71046,N1(C(C(C)OCC)=O)CCC2(CC1)CCN(C(c1cnncc1O)=O)C2 71047,c1(OC)nc(C(=O)NC2CCC(NC(c3cc(Cl)cs3)=O)CC2)cc(O)n1 71048,N1(C(CNC(=O)NC)=O)CCCC(C)(C(=O)NC(c2ccncc2)C)C1 71049,c1(CNC(C(C)OC)=O)ccc(CCNC(=O)CC(C)(C)c2cccs2)cc1 71050,Cc1nc2ccccc2n1CC(N1CC(C(C)NC(c2ccnnc2)=O)C1)=O 71051,CCC(C)(CNC(=O)C(F)C(C)C)C(=O)N1CC(O)(C(C)C)C1 71052,C1(C(C)NC(c2c(CC)ocn2)=O)CN(C(=O)C(C)(C)c2cccs2)CCO1 71053,CCCCC(CNC(=O)C(C)(C)N1CCCCC1)NC(c1cnccc1Br)=O 71054,N1(CC(=O)N(C2CCc3ncsc3C2)CCCCCC)CCc2cc(F)ccc2C1 71055,CCCCC(C)N=c1cc(NCCCCCOCC2CC2)nc(C)[nH]1 71056,c1(NC(C)=O)ccc(C(N2CCC(CNC(=O)Nc3cncc(C)c3)C2)=O)nn1 71057,C1(CC)CN(C(=O)C(=O)NC2CC2)CCC1NC(=O)C(c1cnn(C)c1)O 71058,CC(C)CC(C)CNC(c1csc(-c2ccccn2)n1)=O 71059,N1(C2(C(=O)NCC(CNC(CC=CCC)=O)OC)CC2)CCCCC1=O 71060,C1(C(N(CCC(=O)NOCCC2CC2)CC#C)=O)CC2C=CC1CC2 71061,CS(=O)(=O)C(C(=O)NC1CCC1NC(=O)COCCOCCO)C1CCCCC1 71062,c1(C(=O)NCC(C)(CO)NC(C2C(CCOC)C2)=O)cccc(-c2cnco2)c1 71063,c1(CN(C(C(OC)OC)=O)CCCNC(C2(C)CSC2)=O)ccccc1 71064,C(=O)(CCCC(C)(F)F)NC1(CCOC)CCN(C(=O)C(C)C2(O)CCC2)C1 71065,c1(OCC(N2C3CC(NC(COCC)=O)C2CC3)=O)ccc(C#N)cc1Cl 71066,C1(C(N2CCC(C#CC)C2)=O)CCC2CCC1N2C(c1coc(C)c1)=O 71067,C(=O)(C1=CCC2CCC1N2C(c1coc(C(F)F)c1)=O)NCCCOCCCC 71068,C(=O)(C#CC1CCCO1)N(CCC)CCN(C(C1(OCC)CCCCC1)=O)CC 71069,N1(C(C=CC(C)NC(C2CC(=O)N(C)C2)=O)=O)CCc2cc(F)ccc21 71070,C#CCC(C(=O)NC1COCC1F)NC(c1ccnc(C)c1)=O 71071,N1(C(C(C(C)C)SC)=O)CCCN(C(C2(c3ccc(Cl)c(Cl)c3)CC2)=O)CC1 71072,C#CC(C)(C)C(=O)N1CCC(C(=O)NCCC(=O)NC(C)C)O1 71073,c1(N(C)C)cc(C(=O)NC2CCC2C2CC2)nn1-c1ccc(Cl)cc1 71074,c1(C(N2CCC(C)(C(=O)NCC(C)NC(c3cnco3)=O)C2)=O)ccc(Cl)cc1 71075,C1(NC(c2c(CC)nc[nH]2)=O)CCC(N(C)C(C2CCN(C3CCC3)C2)=O)CC1 71076,Cc1nn(C)c2sc(C(=O)NCCC(C)CCNC(C3CCOC3)=O)cc12 71077,c1(C(=O)NC2CN(C(c3cc(OC)c(F)cc3)=O)C2)cn(C)cc(Br)c1=O 71078,C1(N(C(=O)CC2CCOC2)CCC)CCN(C(=O)Cc2cc[nH]n2)CC1 71079,C1(C(=O)NCC2CC(C)N(C(c3cnc[nH]c3=N)=O)C2)CCCC(C)(C)O1 71080,C1(C(N(CCN(C(=O)CC(C)n2cc(Br)cn2)C(C)C)C)=O)CNC(=O)C1 71081,Cc1sc(O)nc1C(N1CC(F)(C(=O)NC2CCOCC2F)C1)=O 71082,N1(C(c2ccc(-c3ccccc3)s2)C(=O)C=O)CCC(O)CC1(C)C.C(CCC)N.CS 71083,c1(CC(C(=O)CC)N(c2cccc(N(C)C)c2)CC)ccc(F)cc1.OC 71084,CCC(C)C(C(=O)N1CCC(NC(=O)C(Cl)=CCl)C(O)C1)NC(=O)OC 71085,C1(OC)CN(C(=O)C=Cc2ccccc2)C(C)(CNC(c2nncs2)=O)C1 71086,c1(C(=O)NC2CCc3n(C)cnc3C2)ccc2c(=N)[nH]cnc2c1 71087,C1(C(N2CCN(CC(C)NC(c3c[nH]c(=N)o3)=O)CC2)=O)CCCCC1(C)C 71088,C#Cc1ccnc(C(=O)NC(CC=C)C(=O)N2CCOCC2CCO)c1 71089,C1(NC(c2c(NC)nc(C)cc2)=O)CC2CC(C1)N(C(c1cccc(F)c1)=O)C2 71090,C1(C(=O)NCC(=O)OCC=C)CCCC(NC(C2(N(C)C)CC2)=O)CC1 71091,c1(CNC(CC)(C)CNC(c2cccc(CO)c2)=O)cc2cc(C)[nH]c2cc1Cl 71092,C(CC(C)CCNC(=O)CCC1CCCO1)NC(C1N(C(C(C)C)=O)CCC1)=O 71093,C1(NC(C2(CC=C)CC2)=O)CCC(O)CN(C(C2CC23CCSCC3)=O)C1 71094,CCC(CC)C(C(=O)NCCCNC(C1(c2ccccc2F)CCC1)=O)OC 71095,C(C(CN=c1[nH]c(Cl)nc2ccc(Br)cc12)OCc1ccccc1)OC 71096,N1(C(C(COC)C)=O)CCOC2(CCCN(C(c3ccc(CN(C)C)[nH]3)=O)C2)C1 71097,C(=O)(C(C)(C)CC(C)(C)C)N(CC(C)CNC(=O)C1=CCCC1)C 71098,C1(CC)CCC(C(=O)CNC(N2CCC2C(C)C)=O)C1 71099,Cc1cc(C)c(C(N2CCCC(NC(=O)C#CC3(C)CC3)CC2)=O)c(S)n1 71100,C=CCCC(C(=O)OC)N(C(=O)C(CC)OCCCN=[N+]=[N-])CC1CCOC1=O 71101,C1(C(=O)Nc2ncccc2C2CC2)CC(F)CN(C(=O)CC2CCSC2)C1 71102,C=CCC(C(=O)N1CCC1(C)CC(=O)NC1CC(C)C12CC2)OC 71103,c1(-c2n(CCC)ncc2)ccc2c(C(N3CC(O)CC(O)C3)=O)nsc2c1 71104,C1(CNC(c2nc(C(C)(C)C)oc2)=O)CCn2cc(C(=O)O)nc2C1 71105,c1(SC)ncc(C(N2CCC(F)(C(N3CCOC(C(F)(F)F)C3)=O)C2)=O)cn1 71106,C1(NC(=O)CCCCO)C(CNC(C2CN(CC(F)(F)F)C2)=O)CCC12CCC2 71107,CCCC(C)(C)C(=O)N1CC2CC1CC2CNC(c1cccc(=S)n1O)=O 71108,Cc1nsc(N)c1C(N1CCC(CC(=O)NC2CC(CC(N)=O)C2)CC1)=O 71109,C12(C(=O)NCC=CCNC(=O)CC3(O)CCC3)CCCC1C2(F)F 71110,c1(C(N(CC(CN(C(C(CC)F)=O)C)O)C)=O)cnc(OC2CCOCC2)cn1 71111,c1(C(N(CC(C)NC(c2cc(C)ncc2C)=O)CC)=O)coc2cc(C)ccc12 71112,C(=O)(CC(C)CC)NC1(C)CN(C(COCCC#C)=O)C1 71113,Cc1cc(C2CC2)ncc1C(=O)NCC1CCC(C)CN1C(c1cnccn1)=O 71114,C1(CNc2nc(COC)nc(N3CC4CC3CS4)c2)CCC2(CCOCC2)C1O 71115,CC1CCN(C(C2CC23CC(O)C3)=O)CCN1C(=O)CCC1CC1(F)F 71116,N12CCC3(CC3C1)NC(=O)OC1(CC1)CC2=O.N1(CC(C(C)(C)C)=O)CCCC1 71117,N1(C(c2nn(CC)nc2C)=O)CCC(C(N2CC(O)CC2C(N)=O)=O)C(C)(C)C1 71118,CC1C(NC(=O)CSC(C)(C)C)CCCN1C(=O)CN(c1ccc(Cl)nn1)C 71119,N1(C(c2ccc(SC)o2)=O)CCCC(C(C)NC(c2nn[nH]c2Cl)=O)C1 71120,N1(C(C(C)OCOC)=O)CCOC(C)C1C(=O)NCCC(O)C(F)(F)F 71121,c1(C(=O)NC(CNC(c2ccc(NC(=O)OC)cc2)=O)(C)C)nn(C)c(Cl)c1Cl 71122,CCCC(CC)CC(=O)NCC1COCCN1C(=O)CN(C)CC 71123,N1(C(CCc2ccc(C)cc2C)=O)CC2(NC(C3CC3C(F)F)=O)CCC1CC2 71124,N1(C(=O)C=C2CCC2)CCCC2C1CCCCN2C(=O)CCF 71125,C1(C2(O)CN(C(C3CC3C)=O)C2)(CNC(Cn2nc(C)c(Br)c2C)=O)CC1 71126,C1(NC(C=C(C)Cl)=O)CCCN(C(C2CC(C#N)C2)=O)C1 71127,C1(NC(=O)CN2CCCCC2)C=CCN(C(C2(c3ccc(Cl)s3)CCC2)=O)C1 71128,C1(NC(c2cc(C)n(C)c2C)=O)CCC2(CC1)CC(NC(=O)C(F)(F)C(C)O)C2 71129,C(=O)(C#CC(C)(C)CN1CCCC1)NC(c1c(C)nccn1)C1CC1 71130,c1(C(=O)NCC(CO)NC(CC(=O)NCC)=O)csc2c(Br)cccc12 71131,c1(C(=O)NC(CNC(c2c(CC)noc2)=O)(C)CO)ccc(C)c2c1CCC2 71132,N1(C(C2C(C)CC(C)O2)=O)CC2CCN(C(c3ccc(=O)n(C)c3)=O)CCC2C1 71133,Cc1scc(C(N2CC(NC(=O)C(C)(C)C3CCCC3)C(F)C2)=O)c1C 71134,Cc1ncc(C(=O)NC(C)(C)CCNC(C2CC(C3CC3)=NO2)=O)cc1N 71135,C1(C(N2C(C(=O)Nc3cccc(OC)c3)(CC)CCC2)=O)OC(C)(C)OC1(C)C 71136,CCC(O)C(C)(C)C(=O)N1CC(NC(c2cn(CC)nc2C)=O)CC(C)C1 71137,N1(C(C2(Cl)C(C(C)=O)C2)=O)CCOCC(C(N2CCN(C)C(C3CC3)C2)=O)C1 71138,C(=O)(CCCCCNC(c1coc(C(F)F)c1)=O)N1C(C)C(O)CC1 71139,C(C(F)(C(=O)NCCC1CCCC1(C)C)C(C)C)NC(c1nc(OCC)oc1)=O 71140,c1(OC)ccncc1C(=O)NC12CC(NC(=O)C(C)(C)CC3CCOCC3)(C1)C2 71141,CC(C)CCC(O)C(=O)NCCCCCCN(C)C(c1cn(C(C)C)nn1)=O 71142,C1(C)(C(N(CC)CC2CCC2)=O)CNC(C)(C)C1 71143,c1(NCC(CSC)(C)C)cc(=NCC(c2ccsc2)N(C)C)[nH]c(C)n1 71144,c1(C(=O)NCC(CC)NC(c2ncnn2C)=O)noc2cc(F)ccc12 71145,c1(C(N(C(C)C(N2CCN(CCF)CC2)=O)C2CC2)=O)cn(C)ccc1=O 71146,C1(C(=O)NC(C#C)CC)CCN(C(=O)C(C)COC(C)=O)CCO1 71147,C1(C(=O)NCC(C(C)C)OC)(NC(c2cc(O)nc(C)n2)=O)CCC(C)(C)C1 71148,C(=O)(C1CCOc2ccc(Cl)cc21)NC1CN(C(CCC(N)=O)=O)C2(C1)CCC2 71149,c1(C(C(=O)NCC(COC)NC(c2c[nH]nc2C(C)(C)C)=O)C)cccnc1 71150,C#CC1CCCC(CNC(C2(C)CN(C(C3CCC(C)(C)C3)=O)C2)=O)C1 71151,C12(NCc3c(C(=O)OCC)n[nH]c3)CC1CN(C(C1CCC(CC)CC1)=O)C2 71152,C12(C(=O)Nc3n(CC)ncc3)CCC(C(N3CCC(O)C(O)C3)=O)(CC1)CC2 71153,C=CC1(NC(C2N(C(C3CCC3OC)=O)CCC2(C)C)=O)CCOCC1 71154,CC1CCCC(OCC(=O)NCc2cn(C3CN(C(=O)CC4(C)CC4)C3)nn2)C1 71155,c1(C(C(=O)NC(C2CCN(C(C(CSC)C)=O)C2)C)C)ccccc1C 71156,c1(OCC(=O)NC2CC(NC(C(C(C)O)C)=O)C2)ccc(Cl)c(F)c1 71157,Cc1ccc(OCC(C)NC(C2CCN(C3CC3)CC2)=O)c(F)c1 71158,Nc1nc(C(=O)NCC2CC(F)(CNC(=O)C(F)n3cccn3)C2)ccc1O 71159,CCCC(CC(C)C)C(=O)NC1CN(C(c2ccn(C)c2)=O)CCC1O 71160,c1(OC)ccnc(C(N2CCN(C(=O)C(C)n3ccnn3)C(CCO)C2)=O)c1O 71161,c1(C(=O)NC(CNC(c2c(CCC)cccc2)=O)C)ccnc(F)c1N 71162,Cc1csc(C(N2CCC2(C)CC(=O)NC2(CC(C)C)CC2)=O)c1C 71163,C1(C(N(C2CCN(C(C3(C#N)CC=CC3)=O)C2)CC)=O)CCCCC1O 71164,c1(C(=O)NCC2N(C(c3ccc(=O)oc3)=O)CCOC2)c(Cl)cc(Cl)cc1Cl 71165,c1(CNC(C(CO)N(C)C)=O)ccc(C(N2CCC(C)(CO)C2)=O)cn1 71166,C(=O)(C1COc2ccccc21)NCCN(CCC)C(C1(C)CC(F)(F)C1)=O 71167,n1(CC(N2CCC(O)(CN(C(C(C)C(F)F)=O)C)C2)=O)cnc2ccccc12 71168,C(=O)(CC1=CCCCC1)N1CC(C#C)(C(=O)Nc2[nH]ccc(=O)c2C)C1 71169,C(C(=O)NCCCN(C)C)N(CCC)C(C1CC1CSC)=O 71170,CCC(C)CCCC(=O)NC(c1nocc1C(=O)NCC(C)N(C)CCOC)C 71171,c1(C(=O)NCC2C(OC)CCC2)ccc(CNC(=O)CNc2c[nH]c(C#N)c2)cn1 71172,N1(C(C(C)CC(C)(C)C)=O)CCC2(CCCN2C(=O)C(C2CCOCC2)O)C1 71173,CCCCCCN(CC(=O)NCC(CCC)NC(c1coc(SC)c1)=O)C 71174,c1(C(N)=O)ccc(Cl)nc1NC(C1CCCC1NCc1ccnc(O)c1)=O 71175,O(C1CCCc2nc(C)sc21)C(CNC(=O)NCCOC)=O 71176,C(=O)(C(O)C(F)(F)F)OC(C)(C)C.C1(SCC2C(=O)O2)CCCOCCC1 71177,c1(C(N2CC(CNC(C(CN(CC)CC)F)=O)(OC)C2)=O)cccc(F)c1C 71178,CC1CCc2[nH]c(C(=O)NCCCN(C(=O)CC(C)(C)O)C3CCCC3)cc2C1 71179,N1(Cc2cn(CCNC(CCCCC)=O)nn2)CCCN(C(=O)C(C)O)CC1 71180,C1(C)(CCNC(c2c(OC)ccs2)=O)CCN(C(C2(O)CCSC2)=O)C1 71181,C1(C#N)(C(N(CC=CC(=O)NC2CN(C(C)C)C2)C)=O)CC2CC2C1 71182,N1(C(CC)=O)CCc2cc(C(N3CCC(F)C(NC(=O)CSC)C3)=O)ccc21 71183,c1(C(=O)NC2C(NC(c3ccccn3)=O)CCCC2)ccc(O)nc1Cl 71184,N1(C(C2C(C)(C)C2)=O)CC2CCN(C(=O)CCc3cccc(Cl)c3Cl)CC2C1 71185,C(C1C(C(=O)NCC2CN(C(=O)Cn3cnnc3)CCO2)C1(C)C)=C(C)C 71186,c1(C(=O)NC2CC(NC(=O)CC(F)(F)C(F)(F)F)C2)cc(Cl)cc2ccncc12 71187,c1(C(=O)NCC(CNC(=O)CC2C=CS(=O)(=O)C2)OC)ccc2cncn2c1 71188,C1(NC(c2ncc(Br)cc2O)=O)CCN(C(c2ccc[nH]2)=O)C12CC2 71189,c1(C=O)cc(Br)c(C)cc1O.C12(F)CN(C1)N(CCn1cccc1)C2=O.CS 71190,C(C(C)(C)CC(=O)N1CC(CC(=O)NC(c2[nH]c(C)nc2C)C)C2(CC2)C1)OC 71191,c1(C(CCC(=O)NCCOC)=O)c(F)cccc1F.Cc1cc(C(=O)OC)nn1C1CC1 71192,N1(C(C2CC(C#N)(OC)C2)=O)CCOCCC1C(=O)NC1(CF)CC1 71193,S(=O)(=O)(c1ccc(N2CC=C(F)C2)c(F)c1)NCC1OCC(C)C1 71194,C(=O)(C#CC1CCCOC1)N(C1CCCCN(C(C=C(C)C(F)F)=O)C1)C 71195,C1(CC(=O)N(CC#CC)C)CCCCN1C(c1cn(C)nn1)=O 71196,c1(CNC(C(CC)C)=O)ncccc1CNC(c1cc(Br)nn1C)=O 71197,C1(CCC(=O)N(CCN(C)C)C)CN(C(=O)OC(C)(C)C)CCO1 71198,C12(C(=O)N(CCNC(C3(CO)CCCO3)=O)CC3CC3)CCC(CO)(CC1)CC2 71199,CC(C)(C)C(C(=O)NCC1CC1Cl)NC(c1ccco1)=O 71200,c1(C(=O)NC2(CO)CN(C(C3(F)CCCOC3)=O)C2)ccc2nccn2n1 71201,c1(C(=O)NCCCN(C(C)C)C(C2CCC3CC23)=O)ccc2c(c1)CCOC2 71202,CC(CCCNC(c1cccnn1)=O)NC(C1CCCC1c1nc[nH]n1)=O 71203,n1(CC)cnc(C(=O)NC(C)CCN(C)C(c2coc(-c3csc(C)n3)c2)=O)n1 71204,C(=O)(CC(O)CC1CC1)NC(C)(C)CNC(=O)CNC(=O)OC(C)(C)C 71205,N1(CCC)CCC(C(=O)N(CC(C)O)CCNC(=O)CCC2CCC2)CC1 71206,N1(C(C2C(CNC(CNC(CCC)=O)=O)OCC2)=O)CCOCC(C(C)C)C1 71207,c1(C(N2C3CN(C(C4C(C(C)C)C4)=O)CC2CC3)=O)ccc2c(n1)CCC(C)C2 71208,N1(C(CCc2n(C)ccn2)=O)CCCCN(C(c2cccc(OCC#N)c2)=O)C1 71209,N1(C(c2cscc2Br)C(=O)NCCCSCC)CCCC2(CCNC2=O)C1 71210,Cc1nnc2n1CCC(NC(=O)NC(C)(C)C(C(=O)O)c1ccccc1)C2 71211,c1(N2CC(CC(C)NC(c3ccc(CO)nc3)=O)C2)ncc(O)cn1 71212,C1(C(C)C(=O)N(CC(C2CCCC2)O)C)CCN(C(=O)CC2CCSCC2)C1 71213,N1(C(CCN(C(C)=O)C)=O)CC2(CC(NC(=O)C(C)(C)C(C)O)CO2)C1 71214,C(=O)(C(C)Cc1cnc[nH]1)O.C1(C(C2CCCC2)C)CN(C(=O)CN(C)CC)C1 71215,C(=O)(C(O)C(F)(F)F)N1CC2C(CNC(C(CCO)N(C)C)=O)(C2)C1 71216,CCCCC(CNC(C1CC(NC(=O)CC2(OC)CCC2)C1)=O)CC 71217,N1(Cc2c(OC)cccc2C)CCC2(CCN(C(=O)Cn3cc(Cl)cn3)C2)C1 71218,CCCC(CCC)CC(=O)NCC1CN(C(c2ccsc2CC)=O)CC12CCC2 71219,c1(C(=O)NCC(CC(=O)N2CC(n3ncc(C)c3)C2)O)cccc(F)c1C 71220,CN1N=C(C(=O)NC2CCOCC2NC(=O)CC2COC(C)(C)CO2)CCC1=O 71221,N1(C(c2[nH]nc(OC)c2Cl)=O)CC2(CCC2NC(c2ccc(CO)cc2)=O)C1 71222,C1(C(=O)NCC(C)NC(c2c(OC)cnc(Cl)c2)=O)CCOCC12CCC2 71223,c1(C(=O)NC2CC(CC(=O)NCc3c(C)ccc(Cl)c3)C2)cc2cccnn2n1 71224,N1(C(CC2CC(SC)C2)=O)CC2OCCN(C(=O)CCC(=O)N(C)C)C2C1 71225,C1(C(=O)NCCc2cn(C)nc2)CC(NC(=O)Cn2ccnc2)CCO1 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71243,C1(CC(=O)NCCNC(Cc2[nH]c(=N)sc2)=O)CCCC12NC(=O)NC2=O 71244,C(C)(C)(C(C)CC(=O)NC1CC1C1CCC1)NC(C(CCN(C)C)O)=O 71245,C=CCC(C(=O)N1CCCC1COC)NC(=O)CC=C(C)C 71246,N1(Cc2cncc(C)n2)CCC(O)CC1C(=O)NC1CC1c1ccc(Br)cc1 71247,C1(CC#C)(C(=O)NC(CNC(c2cnn(C(C)C)c2F)=O)CO)CC=CCC1 71248,c1(C(=O)NC(CCCC(=O)N(C2C(OC)COC2)C)C)cccn2ccnc12 71249,N1(C(c2c(C)nsc2)=O)CCC2CN(C(=O)C(O)CC3CCCCC3)CC12 71250,C1(NC(COc2cn(C)nc2)=O)CN(C(=O)CN2CCN(C3CC3)C2=O)CC1O 71251,Cc1cc(C(N2CCSCC2C(=O)N=c2cc[nH][nH]2)=O)ccc1F 71252,c1(C(N2CCC(C)C(NC(c3nsnc3O)=O)C2)=O)ccc(C#N)c(Cl)c1 71253,C1(C2CCN(C(c3cc(CO)c[nH]3)=O)CC2)(NC(c2cnc(C(C)C)[nH]2)=O)CC1 71254,N1(C(C=CC(C)C)=O)CC(O)(C(C)NC(=O)CNC(C2CCC2)=O)C1 71255,CCCCCC(CC)C(=O)N1CC(C)CC1C(=O)NOCC1CCCCC1 71256,c12c[nH]c(c1C)C(=O)NC2.N1(C(C(=O)NC(CC)(C)C)=O)CCC(OC)C1 71257,C(=O)(C1CSc2ccccc21)N(C)CCNC(=O)COC(F)F 71258,C1(C(=O)NC(CNC(CN2CC(C)C2)=O)(C)C)CC(c2ccccn2)=NO1 71259,C#CC1(C(=O)NC2CCS(=O)CC2)CCN(C(=O)C(F)n2ccnc2)C1 71260,N1(c2n(CC=C)c(C(C)CC3CCCCC3)nn2)CCC2(CCOCC2)C1 71261,Cc1ccc(C(=O)NC2CCCC2NC(c2scnc2C2CC2)=O)o1 71262,C1(NC(CCCC=C)=O)CCCOC12CCN(C(=O)CC(C)F)CC2 71263,c1(C(N2CC(C3OCCN(C(c4c(C)nns4)=O)C3)C2)=O)cc(Cl)cc(Cl)n1 71264,N1(C(C2(N(C(c3cnn(C(C)C)n3)=O)C)CC2)=O)CC(C)C(C)C1C 71265,c1(-c2c(C)ccc(CO)c2)cnc2[nH]cc(C(=O)Nc3ccnn3CCO)c2c1 71266,CCC(C)C(O)C(=O)N1CCCC1C(C)NC(=O)C=CC=Cc1ccccc1 71267,C1(NC(CC=CC=C)=O)CCN(CCNC(=O)CNC=O)CC1 71268,Cc1ccc(C(=O)NCC2C3CN(C(c4c(C)csc4Cl)=O)CC23)c(O)n1 71269,C12(C(N(C3CN(C(C4(O)CCC4)=O)CC34CC4)C)=O)CCC(C)(CC1)CO2 71270,c1(C(=O)NC(C(CO)NC(c2cc(C)no2)=O)C)cnc2n1CCC(C)C2 71271,C1(CN=C(NCc2cc(C)c(F)cc2)NC2CCOCC2)CCS(=O)(=O)C1(C)C 71272,Cc1cc2cc(C(=O)NC3CC4(C3)CC4C(=O)NC3CCC3)oc2cc1C 71273,C(=O)(C#CC1CCCCO1)NC1CC(C)(C)CN(C(=O)CC(F)(F)F)CC1 71274,c1(C(N(CC(O)CN(C)C(C2CC=CC2)=O)C)=O)ccc2cncnc2c1 71275,C1(CC)(NC(=O)CSS(C)(=O)=O)CCCN(C(c2cncc(OC)c2)=O)C1 71276,C(c1ccncc1)=CC(=O)NCC(C(=O)NC(c1nc[nH]n1)CC)N(C)C 71277,N1(CCNC(C2(CCCC)CC2)=O)CCCN(C(=O)CC2CC2C(F)(F)F)CC1 71278,c1(COC)nc(C)ncc1C(=O)NCC1CCC1NC(c1ccc(CF)cc1)=O 71279,CC(C)(C(=O)NCC1CCN(C(C2(c3cccnc3)CCC2)=O)C1)C1CCCC1 71280,c1(N2CCC(CCNC(C3CC(CCC)OCC3)=O)C2)cc(C)nc(Cl)n1 71281,c1(CNCc2ccc(C3CC(F)(F)C3(F)F)o2)cccc2c[nH]nc12 71282,c1(C(C)C)nnsc1C(C)NC(=O)N(CCCCOC(C)(C)C)C 71283,N1(C(c2occ(S(C)(=O)=O)c2)=O)CC2CCCN(C(c3n[nH]c(=N)s3)=O)C2C1 71284,c1(CCC)cccc(C(=O)NCCC2CCCCN2C(=O)C(C)SC)c1 71285,CCCC(C)(O)C(=O)N1CCC(C)(CC(=O)NCC2(O)CCCC2)C1 71286,N12CC=CC1COCC2=O.C1(C(N2CC(C(=O)OC(C)(C)C)C2)=O)C2COCC12 71287,C1(C(=O)NC2C(C)CN(C(=O)CCc3cncc(F)c3)C2)CCC2C(C1)C2(F)F 71288,CC(C)CC(O)C(C)C(=O)N1CC(F)(F)CC1C(=O)NC1C=CCCC1 71289,C1(C(N2CCC(OCCNC(=O)CSC(F)F)C2)=O)C(C(F)(F)F)C1[N+](=O)[O-] 71290,N1(C(c2cc3ncc(-c4c(C)cco4)cc3[nH]2)=O)CCc2c(Br)cccc2C1 71291,c1(CC)c(C(N2CC3C(CNC(c4n[nH]c(CC)c4Cl)=O)C3C2)=O)csc1C 71292,c1(CC(C)C(=O)NC2(C)CCN(C(C34CC(CN3C3CC3)C4)=O)C2)ccccc1F 71293,C1(CNC(C(CC)N(CC)CC)=O)CC2CCC1N(C(=O)CCCC(N)=O)C2 71294,CCCCCCCC(C)CN=c1[nH]c(=NCC2CCOC2)[nH]c2cc[nH]c12 71295,C1(NC(=O)NCC(=O)NCCC)CC(C)N(C(c2n[nH]c(COC)n2)=O)C1 71296,c1(C(CNC(=O)OC(CC)C(=O)NC)=O)ccc(C)nc1 71297,c1(CC)ncnc(N2CC(C)(C(=O)Nc3cncc(C4CC4)c3)C2)c1F 71298,Nc1c(O)ccc(Cl)c1C(=O)NCC1CCCN(C(=O)C=CC2CCC2)C1 71299,C1(C)(C(=O)NCCN(CCOC)C(c2ccc[n+]([O-])c2)=O)CNC(=O)C1 71300,C(=O)(C(F)(F)C(F)(F)OC(F)(F)F)NCC1(F)CC(CNC(CNC(C)=O)=O)C1 71301,Brc1ccc(C2CCN(CCCCc3nccs3)CC2)nc1 71302,O=S(=O)(c1ccc(Br)c(Cl)c1)Nc1cc(-c2ccc(CCCO)cc2)ccn1 71303,c1(C(=O)Nc2cc(C(C)C)cc(C(C)C)c2O)cnc2c(c1)NC(=O)CS2 71304,c1(C(=O)NC2CN(C(C3(COC)CC3)=O)CC(O)C2)cnc2cc(C)nn2c1C 71305,C1(NC(Cn2c(C)nnn2)=O)CC2CCC1N(C(c1nnc(O)nc1O)=O)C2 71306,Cn1nc(C(N2CCC(NC(C3(CO)CC3)=O)C(CO)CC2)=O)c2c1CCSC2 71307,c1(C(N2CCCC(CNC(C(C)OC)=O)C2)=O)cccc2[nH]ccc12 71308,C1(C(=O)Nc2ccc(-c3cn(CC(COC)O)nn3)cc2)CCCCC1(C)C 71309,C(CC(C)C)(C(=O)NCC(C)n1cncn1)ONC(=O)C1(CCCC)CC1 71310,c1(OC)ncccc1S(=O)(=O)NC1(c2cccc(C(F)(F)F)c2)CCOCC1 71311,N1(C(CCCNC(N)=O)=O)CC2CC1CCC2NC(C1C2C3CCC(C3)C12)=O 71312,Cc1cc(O)cc(=O)n1CC(=O)N(C)CC1CCN(C(C2C=CCC2)=O)C1 71313,n1(CCC(=O)NC2C3(CCC(NC(C=CC)=O)CC3)C2)sc2ccccc2c1=O 71314,C(=O)(C(F)(F)Sc1cnn(C)c1)NCCN(C(=O)Cc1ccn(C)n1)CCOC 71315,C(CCN(C)C(C1(C)CS(=O)(=O)C1)=O)(C(C)C)NC(c1cn(CC=C)nc1)=O 71316,c1(C(=O)NCC2C3N(C(COCC)=O)C(CC3)C2)ccc(Br)c(F)c1F 71317,C1(=O)C(C(C)(C)C)N1.C1(C(N2CC(N(C)C)(C(N)=O)C2)=O)CC2C(C1)C2(C)C 71318,C1(NC(c2ccc(-n3cnnc3)cc2)=O)CCCC(C(=O)Nc2ncc(F)s2)C1 71319,Cc1csc2nc(N(CCCS(N)(=O)=O)Cc3ccccc3)cc(=O)n12 71320,Cn1c(CNCC2(c3ccccc3)CC2(F)F)cnc1Cl 71321,c1(C(=O)OCC)ncccc1NC(=O)OC(C)(C)C.C12CCOCC1NC(=O)C2 71322,c1(C(=O)NCC2(O)CN(C(=O)Cc3cccc(Cl)c3)C2)cccc2oc(O)nc12 71323,N#CCCC(=O)NC(CC(N)=O)c1cn(C2COCC2O)nn1 71324,N1(C(C(C(C)C)NC(C)=O)=O)CCCC2CN(Cc3ccc(Cl)nc3)CC12 71325,C(=O)(CS(=O)CCC(F)(F)F)N1CC(C)(NC(CC2CCN(C)CC2)=O)C1 71326,C#CCC(C(=O)N1CCN(CC(=O)N(C(CCC)c2nn[nH]n2)CC)CC1)C1CC1 71327,C1(CNC(CC(C)C)=O)CN(C)CCN1C(=O)CCc1ccc(Br)s1 71328,C1(NC(c2cccc(OC)c2)=O)CN(C(c2cc(C)ccc2N)=O)CC2(CC2)C1 71329,c1(C(=O)NCC2C(NC(C(C)OCCC(C)C)=O)CCC2)ccc(Cl)c(Cl)c1 71330,N1(C(C(Cc2cn[nH]c2)NC(c2cncc(OC)c2)=O)=O)CCNC(=O)CC1C 71331,c1(C(N2CC(CN(C(C(C)OCCOC)=O)C)C2)=O)n[nH]c2c1CCCCC2 71332,C1(NC(c2c(C(C)C)ncs2)=O)CCCN(C(c2cccnc2CO)=O)C1C 71333,N1(C(c2cnc(Br)n2C)C(=O)Nc2c(C)cccc2)CCCN(C)C(=O)C1 71334,CC1CCSCCN1Cc1cccc(-c2ccc(F)cc2)c1 71335,CC(C(=O)NCCC1CN(C(=O)CCc2nncn2C)CCO1)C(F)(F)C(F)F 71336,C1(OCC)(CNC(c2sc3nccn3c2C)=O)CCCS(=O)(=O)C1 71337,C1(CNC(C2(CC(C)=O)CC2)=O)(CNc2ccncn2)CC12CCC2 71338,CC(C)CC(C(=O)NC1CC(C)OC1=O)NC(C1CNC(=O)O1)=O 71339,C(=O)(C1=CCOC1)NC(C)CC1CN(C(=O)C(C)c2cccs2)C1 71340,C1(NC(C2(CC=C)CN(C(c3cc(CO)oc3C)=O)C2)=O)C2CCC(C2)C1(C)C 71341,CC(CNC(=O)CC1(N2CCCC2)CC1)(CO)NC(=O)CCC1CCC(=O)C1 71342,CC(C)(C)C1=NOC(C)(C(=O)NC2CCN(CCNC(c3ccc[nH]3)=O)CC2)C1 71343,CCCC(F)C(=O)N1CCC(CC(=O)NCC(C2CC2)N(C)C)CC1 71344,N1(C(CCc2cc(C)on2)=O)CCC2CCC(NC(=O)CCc3cnc[nH]3)C1C2 71345,N1(C(C(C(C)(C)C)=O)=O)CC2CC1CCN2C(=O)CSCC(N1CCCCC1)=O 71346,N1(C(=O)CCCC2CCCO2)CCN(C(=O)CCc2cnc(O)[nH]2)C(CO)C1 71347,c1(C(N2CCC(C)CC2CNC(=O)C2CC2)=O)cc(S(N)(=O)=O)ccn1 71348,C1(COC)(NC(=O)Cc2csnc2C)CN(C(C2CC(OC)(OC)C2)=O)C1 71349,C1(CNC(C(C)(C)c2cccs2)=O)CC2(CCN(c3ncc(O)cn3)CC2)CO1 71350,C1(NC(C2CCN(C(CC)=O)C2)=O)CN(C(=O)CN2CCCCC2)CC1F 71351,Cc1c(C(=O)NCC2CC(C)N(C(c3ccoc3Cl)=O)C2)cccc1C#N 71352,C1(NC(=O)COCCOCCO)CCCC(CNC(=O)CC2CCSCC2)C1 71353,c1(C(N(C2CCCN(C(CCNC(COC)=O)=O)C2)C)=O)ccc(S(N)(=O)=O)s1 71354,c1(OCC)ccc(CN(CC(=O)OC)C(=O)COC(CC)CC)cc1O 71355,c1(NC(C2N(C(c3c(C#N)ccc(F)c3)=O)CC=C2)=O)c(O)cccc1[N+](=O)[O-] 71356,c1(C(N2CCC(c3c(C(=O)NCC#N)cccc3)CC2)=O)ccc(Cl)c(O)c1 71357,c1(OC)nccc(C(=O)NC2CCN(C(=O)C(C)Sc3ccc(C)cc3)C2)c1F 71358,C1(C(=O)OC)CC(C)CN(CC2CC2c2ccsc2)C1.C12(CC1)C(=O)N2 71359,O=C1CCCCCN1Cc1cn(CC2C=CCN2C(=O)CC2CCCO2)nn1 71360,N1(C(c2c(CC)n[nH]c2)=O)CC(OC)CC1C(N1CCC(O)(CN(C)C)C1)=O 71361,c1(C(=O)NC(CC(C)NC(C(CC)N(C)C)=O)C)[nH]nc(OC)c1Cl 71362,c1(OC)cccc(OCCN(CC(C)C)C(C2CC(F)(F)C2)=O)c1 71363,CCCCCC(CC)C(=O)OC(C1CCOCC1)COC 71364,N1(c2c(F)cnc(OCC)n2)C2CCC1CC(NC(c1cc(F)ccc1I)=O)C2 71365,Cc1ccc(O)c(CNC(=O)CCN(C(C2CC3CC3C2)=O)C2CC2)c1 71366,N1(C(COC(C)C)=O)CCN(C(C2CCC(N(C)C)C2)=O)C(C(C)(C)C)C1 71367,N1(C(C(CCOC)C)=O)CCCCCC(NC(c2ccnn2C)=O)C1 71368,C1(O)(C(N2CC(NC(CCC3C(C)(C)C3)=O)C(O)C2)=O)CN2CCC1CC2 71369,N1(C(c2cc(C)ns2)=O)C2CCC1CC(NC(c1cncc(N3CCCC3)c1)=O)C2 71370,c1(CC(N2CC(NC(C3N(CCC)CCCC3)=O)C2)=O)cc(Br)ccc1OC 71371,C1(NC(C(CCOC)C)=O)CC2CCC(C1)N2CCCC1CCCC1 71372,C1(OC)(CNC(=O)C(c2cccnc2)C)CCN(C(=O)CC2CCCS2(=O)=O)C1 71373,C#Cc1cncc(NC(=O)CC2CCCN2C(=O)Cc2ccc(C#N)cc2)c1 71374,C12CCC(N1C(=O)OC(C)(C)C)CN2.N1(C(CCSC)=O)CCCC(C)C1 71375,C1(CNC(c2csnn2)=O)(CO)CCN(C(c2occc2C2CC2)=O)C1 71376,Cc1cccc2c1CCOC2C(=O)NC1CCCN(C(c2nn(C)cc2Cl)=O)C1 71377,c1(CNC(N(C(C)C)Cc2cccc([N+](=O)[O-])c2)=O)ccc2c(c1)COCC2 71378,c1(NC(=O)CC2CCN2C(C2COCCO2)=O)cncc(CO)c1 71379,c1(C(N(C2CC(NC(=O)CP(C)(C)=O)C2)C)=O)ccc(-c2ncc[nH]2)cc1 71380,c1(C(=O)NC(CC)CN(C(=O)CC2CC2(C)C)C)cnc(-c2cccnc2)s1 71381,c1(C(=O)NC2CCC(C)N(CC(N3CCCCC3)=O)C2)ccc([N+](=O)[O-])cc1 71382,C(C1CCN(C(=O)C2=CCCCO2)CC1)=CC(=O)NCc1cc2n(n1)CCC2 71383,CCC(O)(CNC(=O)CC(C)(C)NC(=O)C(C)(O)C1CC1)CC 71384,c1(-n2cc(C(CC)O)nn2)ccc(CN)cc1C#N.N12CCC(C(C)(C)C1)C2=O 71385,c1(OC)cccc(C(=O)OCc2cc(Sc3ncccn3)on2)c1 71386,N1(C(C=CCN(CC#C)C)=O)CCN(C(=O)Cc2ccc(SC)cc2)C(C)C1C 71387,N1(C(C(C)C2CC2)=O)CC2CCN(C(C34CCC(C(F)F)(CC3)C4)=O)CC2C1 71388,c1(NC(=O)NC(c2ccc(Cl)cc2OC)CC)ncnc2c1c(Br)nn2C 71389,c1(N2CC(C(C)NC(CC3C(C)C3)=O)C2)nc(Cl)nc2[nH]ccc12 71390,C(c1nccs1)=CC(=O)NCC(C1CCCC1)NC(=O)COCc1nc[nH]n1 71391,C1(C)(CNC(CS(=O)(=O)N(C)C)=O)CCCN(C(C2CCCC(C)(C)O2)=O)C1 71392,C1(CNC(C(CC)=CC)=O)C2CCC(C2)N1C(=O)CCC1CCCC1 71393,C12(C(=O)NC3CC(CCNC(CNC(=O)OC)=O)C3)CCCN1CC(O)C2 71394,CS(=O)CC(=O)N1CCCC1CNC(c1cc(C(C)(C)O)on1)=O 71395,C1(C(=O)NCCC2(C)CCN(C(CSCC)=O)C2)CCc2nc(C)nn2C1 71396,C(=O)(CC(CC)C(C)(C)C)NC1C(CCC)CN(C(c2cn(C(C)C)cn2)=O)C1 71397,C1(C(C(=O)NC(C(C)C)CN(CC(=O)N(C)C)C)C)CCCC(F)(F)C1 71398,C1(CCCNC(C2(C(C)(F)F)CC2)=O)CCN(C(c2ccncc2O)=O)CC1 71399,C12(CN(C)C(=O)NCc3cnn(C)c3)CCCC1OCC2 71400,c1(CNC(=O)NC(C2COCCO2)C(=O)O)ccc(Br)cc1[N+](=O)[O-] 71401,n1(CC)nc(C(=O)NCCOCCNC(c2cnccc2Br)=O)ccc1=O 71402,c1(OCC(N2CCC(C)(CNC(COCCCOC)=O)C2)=O)ccc(F)c(F)c1 71403,C(=O)(CCP(C)(C)=O)NC(C(C)C)C(=O)NCCC1(C)CCCO1 71404,n1(CCCOC)nnnc1C(c1cc(C(F)F)on1)NCC1(F)CCOC1 71405,c1(CC(=O)NC(CNC(Cn2c(C(C)C)ncc2)=O)C(C)C)ccccc1Cl 71406,C1(CNC(CC(C)N(C)C)=O)CCC2(CO1)CC(NC(=O)CCNC(N)=O)C2 71407,C1(C(=O)NCc2cc(CO)ccn2)CN(C2CC2)CCC1C(F)(F)F 71408,C1(C(=O)Nc2c(C)n(C(C)C)nc2)CCN(C(C2CCC(F)(F)C2)=O)CC1O 71409,c1(NC(=O)NC2(c3ncccc3F)CCOCC2)ccc(C2CC(F)(F)C2)cc1 71410,c1(C(=O)OCCc2ccc(C#N)cc2)ccc(S(=O)(=O)CCS(C)(=O)=O)cc1 71411,c1(OCC)cc(C(=O)NCC(C2CCC2)NC(=O)C2=CCSC2)ccn1 71412,Cc1cc(C(N2CCCC2(C)CNC(=O)CC2CNC(=O)C2)=O)c2[nH]cnc2c1 71413,c1(C(=O)NC(CCNC(Cc2ccc(C)cc2C)=O)C)c(C)nn2ccccc12 71414,CC(C)(CS(C)(=O)=O)C(=O)N1CC2(CCN(C(c3ccc([N+](=O)[O-])cc3)=O)C2)C1 71415,C=CC1CCCCN1C(C1(C)CCN(C(c2nnn(C)c2C)=O)CC1)=O 71416,Cc1noc2ncc(C(N3CCC(N(C)Cc4nc(C5CC5)nn4C)C3)=O)cc12 71417,C(=O)(C(C)(C)C(O)C(C)C)N(CC(=O)NC(CF)CF)CC 71418,c1(OC)cc(C(N2CCSCC2C(=O)Nc2cccnc2Cl)=O)nn1C 71419,c1(C(N(CCN(C(C(C(C=C)C)C)=O)C)C)=O)ccc2c(=N)[nH]cnc2c1 71420,Cc1cc(C(=O)NCC2(C)CCCN2C(=O)CC(C)C2CCCC2)c(O)nn1 71421,CC1(C)CN(C(=O)CC2=CCCC2)CC(CNC(c2cc3c[nH]nc3s2)=O)O1 71422,CC1=CCC=CC1C(N1CCC(CCNC(C2CCCN2C)=O)CC1)=O 71423,N1(C(c2nc[nH]n2)CC)CCc2cc(F)c(F)cc2C1 71424,c1(C(=O)NC2C(NC(CCNC(=O)OCC)=O)C2)c[nH]c2cccc(F)c12 71425,C=C1CCN(C(=O)CCCCOCC)C(C(=O)N(C(CC)CO)C)C1 71426,C1(NC(=O)CC2CCCCC2)CN(C(=O)C(F)n2cccn2)C2CCCCC12 71427,C1(C(=O)NC2CC(O)(CNC(c3c(C)scc3)=O)C2)CCc2nncn2CC1 71428,c1(CN(C)CC2CCCN(C(c3ccc(Br)c(Br)c3)=O)C2)ccc(F)c(F)c1Cl 71429,N1(C(C)C)CCCC1CC(=O)NC1CCCC1NC(=O)C(C)(C)c1ccnn1C 71430,N1(C(Cc2n(C)nnc2)=O)CCCOC(CNC(=O)CN2C(=O)CNC2=O)C1 71431,CC1(C)CC(=O)NCC1C(N1CCC(OCCNC(C2CC(=O)N2)=O)C1)=O 71432,N1(C(C=Cc2n(CC)ccn2)=O)CC2CCC1CN2C(C1CS(=O)(=O)CCO1)=O 71433,N1(C(CC2ON=C(CC)C2)=O)CCCCCC1C(=O)NCCc1cnc(C)[nH]1 71434,C12(NC(c3ncn(CC)c3)=O)CCCC1N(CC1CCCCO1)CC2 71435,C(=O)(CC(C(F)(F)F)NC(C1CC2CC2C1)=O)N(CCCCOC)C 71436,N1(c2ncc(CC)cn2)CCC(NC(c2[nH]nnc2C)=O)C(C)(C)C1 71437,CC1CC(N(C(=O)C(c2ccoc2)NC(=O)COCCCN=[N+]=[N-])C)CCO1 71438,N1(C(c2c(NC)cccc2OC)=O)CC2(CCCN2C(C2(C)CCCCC2)=O)C1 71439,c1(-n2c(C(c3cc(=NC)[nH]cc3)NCCC(F)F)nnn2)ccc2c(c1)CCC2 71440,C1(C(=O)NC(c2cc(F)cc(F)c2)CCOC)CCC(O)C(O)CC1 71441,N1(C(CCC(C)(C)C)=O)CCC2(CCC2NC(c2csc(C(F)F)c2)=O)CC1 71442,C(=O)(C1CCCc2nncn21)NC1CCCCN(C(c2c(=N)[nH]cnc2)=O)C1 71443,C12COCCN(C1)C2=O.C1(C)(NC(C=CC(=O)N(C)C)=O)CCC1 71444,n1(CC)cnc2nc(N3CCC(C)(CC)C3)nc(NCC3CC(C(F)(F)F)C3)c12 71445,N1(C(c2cncc(C)c2)=O)CCC(C)C(N(C)C(c2cn(C3CC3)cn2)=O)C1 71446,Cc1cc(=NCCCCC(C)NC(c2ccc3c(c2)COB3O)=O)[nH]c(CO)n1 71447,N1(C(C2(C)CCCC2)=O)CC(NC(C2(Cc3cnn[nH]3)CCC2)=O)C(CO)C1 71448,C1(NC(CC2CC(=O)NC2=O)=O)CCCN(C(c2nc(F)ccc2Cl)=O)CC1 71449,N1(C(c2cc(C)nn2C)=O)CCC(CCNC(=O)C(O)CC(C)C)C(F)(F)CC1 71450,c1(C(N2C(C(=O)NC(CC)C(C)O)CC(O)C2)=O)cc(F)cc(Br)c1F 71451,CCN=c1[nH]cc(C(=O)NC(C)(C)CNC(=O)Cc2ccc(OC)cc2F)s1 71452,c1(CNC(CC(C(C)C)O)=O)cnn2c1CN(C(c1cncc(O)c1)=O)CC2 71453,C12CCC(CC1)C(c1nnnn1C)NC2CCO.C1(C(F)(F)F)(CC)CCCC1 71454,C1(C)(NC)CN(C(=O)CCC2CCC(NC(=O)C(C)OCC(C)C)C2)C1 71455,c1(CC)nc(C(=O)NCC2CCN(S(=O)(=O)C(F)F)C2)c(Br)s1 71456,C#CCCCCC(=O)N1CC(OC2CCN(C(=O)CC(C)O)CC2)C1 71457,C1(C(N(CC(=O)NC2CC23CCC3)C2CC2)=O)CC(C2CC2)=NO1 71458,Cc1cccc(Cl)c1C(=O)NC1CS(=O)(=O)CC1NC(C1CC2(C1)CC(C)C2)=O 71459,c1(C(=O)NCC2OCCC(NC(C3C(C)C3C)=O)C2)ccnc2c1CCC2 71460,N1(C(C2CS(=O)C2)=O)CC2CCC2(C(=O)Nc2ccc(O)cc2Cl)C1 71461,c1(CN2CCC(C(N(CCC(=O)OC)C3CC3)=O)CC2)cc(Br)c(O)c(Br)c1 71462,Cc1ccccc1-n1nnnc1C(c1nnc(CF)o1)NCCCNS(N)(=O)=O 71463,C1(CNC(C2C(C=C(C)C)C2(C)C)=O)C2CCC1CN(C(c1cc(C)[nH]n1)=O)C2 71464,N1(C(=O)CCc2cccnc2F)CCCN(C(=O)CCC2CCOCC2)CCC1 71465,c1(C(=O)NC)ccc(C(=O)NC2CC2NC(c2cccc(C)c2C)=O)cc1F 71466,[N-]=[N+]=NC1CCN(C(=O)C(CC2CCC2)NC(=O)Cc2cn[nH]c2)CC1O 71467,C(c1ccc(F)cc1F)=CC(=O)NC(C(C)NC(=O)CC(C)(C)O)CO 71468,c1(OC)ccc(C2(C(=O)NCCCN(C(=O)C=Cc3cncs3)C)CC2)cc1 71469,C(CN=c1[nH]c(=NCC(CC(C)C)N2CCC2)[nH]c2c1CCC2)n1ncc(C)c1 71470,C1(C(=O)NC)CCCCN1C(CCC)C(=O)NCc1ccc(OC)cc1 71471,c1(CC)nnc(=NCC2(F)CC(N(C(C3CCCC4CCCN34)=O)CC)C2)[nH]c1CC 71472,c1(CN(C=O)Cc2c(OC)c(F)c(F)cc2)cccc2c1OC(C)(C)C2 71473,N1(C(CC(CNC(c2cc(CCC)[nH]n2)=O)C)=O)CC(=O)NCC12CC2 71474,C1(NC(CCC=C(C)C)=O)CCCCN(C(C23COC(CF)(C2)C3)=O)C1 71475,C1(COC)(NC(C2CCSC2)=O)CCN(C(=O)CCCSC)C1 71476,C1(C(=O)NC2CC(C)(CC(=O)NC(CC#C)C(=O)OC)C2)CCCC2(CC2)C1 71477,C(=O)(CCC(=O)N1CCN(C(=O)CCC2NC(=O)NC2=O)CC1)N(CC)CC 71478,N1(C(CCN(C(=O)CC2(COC)CC2)CC)=O)CC(=O)N(C)C(=O)C1 71479,C(c1sc2ccccc2c1Cl)=CC(=O)N(CC(O)CN=[N+]=[N-])C 71480,N1(C(c2cc(Cl)sc2Cl)=O)CC2CCN(c3ncc4[nH]ncc4n3)C2C1 71481,C(=O)(CCC(C)C)NC12CC(CNC(C3(CC)CCCO3)=O)(C1)C2 71482,N1(C(C=NOC)=O)CC(NC(=O)CSC(C)C)CC(C)C1 71483,C1(NC(C2(C)CCC(F)(F)CC2)=O)CN(C(=O)C(N)=O)Cc2nccn2C1 71484,Cc1cnc(N)c(C(=O)NC2CCC(C)N(C(c3coc(Br)c3)=O)C2)c1 71485,C=CC1(C(=O)NCC2CN(C(=O)C(O)CCN(C)C)CCN2C)CCCCC1 71486,C1(C(N2CC(C)(CNC(c3c(C)nn(C)n3)=O)OCC2)=O)C2CCC3C(C2)CC13 71487,Cc1ccsc1CC(=O)NC1CCC(N(C(=O)Cc2nccn2C)C)C1 71488,CC1(N=c2[nH]c(Cl)nc3ccccc23)CC(NC(c2c(Cl)ccc(F)c2Cl)=O)C1 71489,CC1CC(NC(C23CC4CC2C3C4)=O)CN(C(=O)C(C)Cn2ccnc2)C1 71490,c1(OC)cc(N2CC3CC2CN3Cc2cccc(Br)c2Cl)nc(OC)n1 71491,N#CC1(C(=O)NC(CO)C(F)F)CC12CCOCC2 71492,N1(C(CSCCC(C)C)=O)CCCC(O)(CNC(=O)CCC2CCCN(C)C2)C1 71493,C1(C(=O)Nc2ccc(OC)nc2)(OC)CCN(C(=O)CC2CCCSC2)CC1 71494,CCC(CN(C)C)CC(=O)NC1CCC(CNC(C2CCN(C3CC3)C2=O)=O)C1 71495,n1(COC)ccc(C(=O)N(CCCCN(C(=O)CCCSC)C)C)n1 71496,c1(CNC(C(C)Cn2cccn2)=O)ncc(C(=O)NCC(CO)N(C)C)cn1 71497,Cc1c[nH]c2ncnc(N3CCC(O)C(C(=O)Nc4ccc(S(C)=O)cc4)C3)c12 71498,CC(Cn1cccn1)C(=O)NCc1cc(C(=O)NCC(O)C(N)=O)cs1 71499,C1(CNC(c2n(Cc3nnn(C)n3)nnn2)c2nc(CO)cs2)CCOC1(C)C 71500,n1(C2CCN(C(=O)C(O)CF)CC2)cnc2c1CCN(C(C1CC(F)C1)=O)C2 71501,C1(C(C)(C)NC(C(C)SC(F)(F)F)=O)CCN(C(=O)CC2COCCN2C)CC1 71502,CCC(CC)C(=O)NCc1cccc(C(=O)NCc2ncnn2C(C)C)n1 71503,N1(C(C(CNC(c2ncccn2)=O)CC2CC2)=O)CCCC2COCC12 71504,C1(CC=C)(NC(CC=CC=C)=O)CCN(C(c2cnc(NC)cn2)=O)CC1 71505,Cc1noc(C)c1C=CC(=O)NC1CCCN(C(c2ccn(C(F)F)n2)=O)C1 71506,C1(C2CC2)(CNC(CCc2ncn(C)c2)=O)CCN(C(c2cnn(C)c2)=O)C1 71507,c1(C(=O)NCC(C2CC2)NC(C(c2ccc(N(C)C)cc2)C)=O)cc([N+](=O)[O-])n[nH]1 71508,N1(C(C(C)OCCN(C)C)=O)CC23CCCCC2(C1)CN(C(=O)C(N)=O)C3 71509,c1(NC(C2CN(C(c3c(Br)cnc(C)n3)=O)C2)=O)ccc(C#N)cc1I 71510,N1(C(C(CCCC)C)=O)CCCN(C(c2ccc(CN3CCCC3)o2)=O)CCC1 71511,CCCC(CCC)CC(=O)N1CC2(NC(c3cc(CC)c(C)s3)=O)CCC1CC2 71512,c1(C(C)(C)C)ccc(CN2CCC(F)(C(=O)Nc3c(Cl)cnn3C)C2)c(F)c1 71513,c1(C(=O)NCC2C3N(C(CN(CCC)C)=O)C(CC3)C2)c(C)ccc(Cl)c1F 71514,CSC1=C(C(=O)N(C(C)CN(C)C(C2(C#N)CC2(C)C)=O)C)CCCC1 71515,N1(C(C=C(CC)CC)=O)CCC=C(C(=O)N2CC(Cc3ccco3)C2)C1 71516,N12CCN(CC1)NCCC2.N1(CCC)CCCC1CCCO.C(C)=O 71517,c1(C(=O)NC2CC3(C(NC(CC4(OC)CC4)=O)C3)C2)csc2nccn12 71518,C1(C(C)NC(c2nscc2Br)=O)CN(C(=O)C(F)=C2CCCC2)CCO1 71519,Cc1nsc2ncc(C(N3CC4CCN(C(=O)CCc5nncs5)CC34)=O)cc12 71520,C(C(C)(C)CC(=O)N1CC=CC(O)C1)NC(C(C)OCC1CC1)=O 71521,C(=O)(C1=NN(c2ccccc2)C(=O)CC1)NCC1N(C(C2ON=C(C)C2)=O)CC1 71522,c1(C(=O)NCCNC(C(=O)NCCC(N)=O)=O)cc(CC2CC2)on1 71523,N1(C(C(C)OC)=O)CCC(C)(NC(=O)CC(C)CNC(=O)OC(C)(C)C)CC1 71524,N1(C(C(CC(C)C)ONC(=O)C=Cc2cocn2)=O)C(CO)CCC12CCC2 71525,C(=O)(C(C)(C)C(O)c1cc(Cl)cc(Cl)c1)N1CC(CC=C)(NC(C2CC2C)=O)C1 71526,C1(N2CC3C(C)C3C2)CCCN(CC(=O)OCCO)C1=O 71527,c1(C(=O)NC2CC2C(=O)NC2(c3ccc(Cl)cc3)CC2)ccc(O)c(Cl)c1 71528,C(CC(C)(C)C(=O)NC(c1ccc(F)cc1)C)NC(c1cnc(C)s1)=O 71529,Cc1nc(S)nc(C)c1CCC(=O)NC(CNC(C1CC(C#N)C1)=O)CC(C)C 71530,C(CCC(=O)NC(c1ccoc1)C)(C(C)C)NC(c1cc(OC)n[nH]1)=O 71531,c1(CC)cccc(C(=O)NCC2CCC(NC(C3(CCOC)CC3)=O)C2)n1 71532,C12(C(=O)NCC(c3ccccc3)CNC(=O)Cc3ccco3)COCC1C2(F)F 71533,C(=O)(C(C)C(O)CC(C)C)N1CC(C(=O)NC23CCN(CC2)C3)(CC)C1 71534,C12(CNC(CNC(C)=O)=O)CC(NC(=O)COCC(F)(F)F)(C1)C2 71535,CCCCN=C(NCC1CCCCC1)N1CC(C)(C)OC2(CCOC2)C1 71536,c1(C(=O)NC(CC)CNC(C2(CO)CCCO2)=O)cc(C)cc2c1NCCC2 71537,O(NC(=O)C#CC(C)(C)CNC(c1cc(F)ccc1O)=O)CCCC=C 71538,C=Cc1cc(C(N2CC3C(NC(c4cnc(S)n4C4CC4)=O)C3C2)=O)cc(F)c1 71539,n1(CC(=O)NC2CCN(C(CC(C)C)=O)CC2(C)C)cnc2c(cnn2C)c1=O 71540,c1(C(=O)OC)ncc(C(=O)NCCN(C(=O)CCc2cc[nH]n2)CC(C)O)s1 71541,N1(C(c2ncccc2Br)=O)CC2CCC1CN2C(c1cccc2c1CCC2)=O 71542,c1(C(C(=O)NC2(c3cc[nH]n3)CC2)N(C)CC2CC2)cc(Cl)cc(Cl)c1 71543,Cc1noc(C)c1CC(=O)NC1CCC1NC(C1COC(=O)O1)=O 71544,C1(CN)CCCC(Nc2ccnc(CNC(=O)C(F)=CCCF)c2)CC1 71545,N1(CC(C)(C)OC)CC(c2ccccc2Cl)OCC1C 71546,C(=O)(C1Cc2ccccc21)NC1CCCCN(C(Cc2cc(C)cc(F)c2)=O)C1 71547,C1(C(=O)NCC2(C)CCN(C(CCCc3ccc(C)s3)=O)C2)Cc2nccn2C1 71548,N1(C(c2ncnc3c2CCC3)=O)CCCC2(C1)CN(C(C1CCCCS1)=O)C2 71549,N1(C(c2c(C)ccc(F)c2N)=O)C2CCC1C(C)C(NC(=O)C1=CCCC1)C2 71550,C1(C)(NC(C(C)N(C(C2(C(C)(C)O)CCC2)=O)C2CC2)=O)CN2CCC1CC2 71551,c1(OC(C(N2CCCC(COC)C2)=O)C)ccc(CNC)cc1 71552,C(=O)(C1(C)OCCc2ccccc21)NCC1C(NC(c2ccn(C)c2)=O)CCC1 71553,c1(C(N2CC(CC(=O)N(CCOC)CCF)C3(C2)CC3)=O)cc2cc[nH]c2cn1 71554,N1(C(c2cc(CC(C)C)on2)=O)CC(NC(=O)CC(C)n2cccn2)CC(C)C1 71555,Cc1cn(C)nc1C(=O)NCc1nc(C(=O)Nc2cncc(F)c2)c(C)o1 71556,N1(C(C(CSC)OC)=O)CCN(C(c2cc(Cl)cn2C)=O)CC(O)C1 71557,C(=O)(C(C(CC)CC)NC(c1occc1CC)=O)NC(CC=C)CC(=O)OC 71558,C1(C)([SH]=CC(=O)N(C)CC2N(C(C3CCC(C)O3)=O)CCCC2)NC(=O)NC1=O 71559,N1(C(CC(CCSC)O)=O)CC2(C1)CN(C(c1nocc1C(C)C)=O)CC2CO 71560,CCCCC(O)C(C)C(=O)NC12CC1CN(C(c1cc(O)ccc1C)=O)C2 71561,C(CCCCN=c1[nH]c(-n2cccn2)nc(=N)[nH]1)N(S(C)(=O)=O)C 71562,CC(CO)C(=O)NC1CC(F)(CNC(=O)CC=CCNC(=O)OC(C)(C)C)C1 71563,c1(N2CCCC(NC(C(C)(C)n3cnnn3)=O)CC2)nc2ccc(F)cc2s1 71564,C1(C(C)NC(c2cnn(-c3nccs3)c2)=O)CCCN(C(=O)C(C)(C)C)C1 71565,C(=O)(C1=C(C#N)CCC1)C(Cc1n(C(C)C)cnn1)=O.C1(CN)C(C)CCCN1 71566,C1(C)(C(N2C(C)CC2C(=O)NC23CC(F)(C2)C3)=O)CC(C)(C)C1 71567,C=C(C(=O)NC1CC(NC(c2cc(Br)ccc2Br)=O)C1)C(F)(F)F 71568,c1(C(CNC(C2(CCOC)CC2)=O)NC(c2cnc(CC)[nH]2)=O)ccc(C)cc1 71569,C1(C2CCN(C(c3ncn(C)n3)=O)C2)(NC(c2ncn(C)c(=O)c2)=O)CC1 71570,C1(C(N2CC(OC)C2)=O)CCC2(CC2)N1C(=O)CN1CCNC1=O 71571,C1(NC(=O)Nc2c(C)sc(C(C)N)n2)CC1C1CCOCC1 71572,Nc1cc(C(N2CC3CC2CC3CNC(C2CCCCS2)=O)=O)cnc1N 71573,C1(C(=O)NC2CC(C)(NC(CC3CCCC(OC)C3)=O)C2)CN2CCN1CC2C 71574,N1(C(c2cc(=O)cc[nH]2)=O)CCC2(CCCN2C(C2CCC=CO2)=O)C1 71575,c1(NC(C2C=CC(NC(=O)CCc3ccc(F)cc3)C2)=O)ccc(Cl)cc1F 71576,C1(NC(CC=C)=O)CC(F)CN(C(=O)Cc2n[nH]c(=N)s2)C1 71577,N1(C(C2N(C)CCOC2)=O)CCN(C(=O)CCN2C(=O)CCC2=O)C(C2CC2)C1 71578,Cc1cc(NCC2(C)CCCCO2)c(Br)cc1[N+](=O)[O-] 71579,c1(C(N2CC(C(=O)OC3C(CCC)C3)C2)=O)cc(CNC(C)(C)C)on1 71580,N12CCC(C1(C)C)CC2=O.N1(C(COCCCCC)=O)CC(O)CC1CO 71581,C1(Cn2cc(-c3nccc(C)n3)nn2)C2CCC(C2)N1C(=O)C(C)C(C)(C)C 71582,C1(O)(N(C(CNC(=O)OC)=O)CCO)CN(C(=O)C(C)(O)n2cccn2)C1 71583,N1(C(C2CCN(C)CC2)=O)CC2CCCC1(CNC(c1cc3cscc3s1)=O)C2 71584,N1(C(C(CCC)OCC)=O)CC2(CCN(C(C3CCCS(=O)(=O)C3)=O)C2)C1 71585,N1(C(CC2(C)CN(C(c3cccc(O)n3)=O)C2)=O)CCCN(CCO)CC1 71586,CC(CC1CC1)C(=O)NCCC(=O)N(C)Cc1ccsc1 71587,C(=O)(CC(F)(F)CC(=O)N1CCOCC1c1nc2ccccc2s1)OC 71588,N1(C(CC(c2ccc(F)cc2)C)=O)CCN(C(c2ccnnc2S)=O)CC1CO 71589,C1(N(C(CCCC(C)=O)=O)C)CCN(C(C2CCC(C)=C(C)C2)=O)CC12CC2 71590,C(=O)(CC(C)C(=O)N1CC2C(NC(c3cnc4sccn34)=O)C2C1)OC 71591,Cc1ccc(C(=O)NC2CN(Cc3ccc(F)c(F)c3)CC2F)c2ccccc12 71592,Cc1cnc(CNC(C2(NC(=O)Cc3ccc[nH]3)CC2(C)C)=O)cn1 71593,C(=O)(C(C1CC1)N(C1CC1)OC(C(=O)Cc1ccsc1)=O)NCCCC 71594,c1(CC(=O)NCCC(=O)NC(C(C)C)C(C)NC(=O)CO)ccc2nn[nH]c2c1 71595,C#CC1CN(C(=O)COCC)CCN1C(=O)CC(C)C(C)C 71596,C(=O)(C(CNC(=O)C(OC)OC)C(C)(C)C)Nc1c(OC)cc(C)cc1 71597,Cc1ncnc(O)c1C(N1CCC(C)(CCNC(C2CC=CC2)=O)C1)=O 71598,C1(C(=O)NC2(C(=O)NCC#C)CC2)CC(C)(C)CCN1C(=O)CC1C=CCCC1 71599,n1(C(C)C)ncc(C(=O)NCC(O)CNC(c2sccc2C(C)(C)C)=O)c1N 71600,c1(C(=O)NCCCNC(C(CC=C)CC)=O)ccc(N)c2ccncc12 71601,CC1CN(C(=O)NCc2cccc3ncnn23)CC2(CCCC2)O1 71602,CCC1=NOC(CC(N2CCC(C(C)(C)CNC(=O)C3=COCC3)CC2)=O)C1 71603,c1(NC(CCCOC)c2cccnc2)cc(Br)ccc1S(=O)(=O)NC1CCCOC1 71604,C1(NC(CNC(=O)OC)=O)CN(C(=O)C(C2CCC2)SC)C2(CCOC2)C1 71605,CCCC(CC)CCC(=O)N1CC(C)(C)CC1C(=O)NCC1(OC(C)C)CCC1 71606,CCCC(C(=O)N1CCCCC1C1(NC(C2(S(C)(=O)=O)CC2)=O)CC1)NC(C)=O 71607,N1(C(Cc2cc(C)sc2)=O)CC(NC(C2CC(C)C2)=O)C(C)C1 71608,c1(C(=O)NC2C(CNC(=O)CC3CCCCO3)CCC2)ccc2c(n1)CCCC2 71609,C1(C(=O)NCC2N(C(COC3C(C)CCCC3)=O)CC=C2)CN2CCN1CC2 71610,N1(C(c2c(CC)ccs2)=O)CC2CC1CCC2NC(c1c[nH]nc1C(C)(C)C)=O 71611,C1(NC(C2C(C)(C)C2)=O)CC2CCC1CN(C(C1(C)CC3CCC1O3)=O)C2 71612,N1(C(=O)CSC(F)(F)F)CCC2CC12C(=O)Nc1cccc(OCF)c1 71613,c1(C(=O)NCC(C)(F)CNC(C2CC2F)=O)cnc2n1CCCC2 71614,Cc1n[nH]c(C)c1C(=O)NCC(CO)NC(=O)C(C)OCc1ccncc1 71615,c1(C(=O)NCc2ccoc2C(=O)NOC2CC3CCC2C3)ccc(O)cc1 71616,C1(CC)CC(C(=O)NC2CCN(c3nnc(COC)s3)CC2)CCO1 71617,C1(NC(=O)C=CCO)CC2CCC(C1F)N2C(=O)CCN1CCC1 71618,O=C(NNC(=O)C1CCS(=O)(=O)C1)c1cncc(OCC(F)F)c1 71619,N1(C(CC=CCC)=O)CCc2ccc(C(N3CCCC4OCCC34)=O)nc2C1 71620,c1(N2CC3CC(NC(C45C(C)(C)C(CC4)C5)=O)CC3C2)nc(Cl)nc2[nH]ccc12 71621,c1(C(N2C(C)(CC(=O)N(c3c(OC)cccc3)C)CC2)=O)cc(F)ccc1O 71622,CC(C)C(N=[N+]=[N-])C(=O)N1CC(OC2(C(C)NC(C)C)CC3CCC2C3)C1 71623,CC1C(C(=O)N2CCC(C(N3CCCC(N=[N+]=[N-])C3)=O)(CO)C2)=NOC1C 71624,C1(CN(C(=O)COCC(C)(C)C)C)CCCN(C(C23CCCC2C3)=O)C1 71625,c1(OC)cc(CCC(=O)NC(C)C(C)NC(c2cc(Cl)c[nH]2)=O)ccc1O 71626,C(=O)(CC(C)C(F)(F)F)NCCNC(CC1(CC(=O)OC)CCCC1)=O 71627,N1(C(Cc2c(C)con2)=O)CCN(C(c2csc(S)n2)=O)CCC1C 71628,N1(C(C2N(C(C)C)CCC2)=O)CCC(F)(CNC(=O)C(C)c2cccs2)CC1 71629,C1(NC(c2ccc(C(F)(F)F)o2)=O)CCC2(CCN(C(c3ccon3)=O)C2)C1 71630,C(=O)(C(O)CC(F)(F)F)NCC1CN(C(COCc2scc(C)c2)=O)C(C)(C)C1 71631,C#Cc1ccc(C(=O)N(C(C)CCNC(C23CCC(CC2)O3)=O)C)c(F)c1Cl 71632,C1(NC(=O)CCNC(=O)Cc2cscn2)CN(C(C2CCC2)=O)CC1C1CC1 71633,N1(C(CC(CNC(c2cn(CC)nn2)=O)OC)=O)CCC2(CCCCC2)C1 71634,n1(CC(N2C(CCNC(CCNC(=O)NC)=O)CCC2)=O)ccc(C)cc1=O 71635,CCN=c1[nH]c(C(N2CC3C(CNC(=O)COC4CCN(C)CC4)C3C2)=O)cs1 71636,C1(NC(C2OCCN(CC)C2)=O)CCN(c2nnc(C3CC3)o2)CC1F 71637,c1(CC)ccc(C(N2CCOC(CCOC)CC2)C(=O)NCCSC)cc1F 71638,O([Si](C)(C)C(C)(C)C)Oc1sccc1C(N1CC(C(=O)OC)C(F)C1)=O 71639,Cc1cc(=NCC(O)CNC(C2CCS2(=O)=O)=O)[nH]cn1 71640,Cc1cc(C(=O)NCC2CCN(C(C3C4CCC(=O)C34)=O)CC2)cc2c1CCC2 71641,N1(CCNC(N2CCC(CN)CC2)=O)C(=O)NC2(CCC2)C1=O 71642,c1(C(N2CCC(C)(CNC(C(C(=C)Cl)(C)C)=O)C2)=O)cccc2nn[nH]c12 71643,c1(C(=O)NCCC(CNC(c2ccc(C)nc2O)=O)O)cccc(C=C(F)F)c1 71644,c1(C(=O)NC(C)CNC(=O)Cn2ncnn2)nccc2c(Cl)cccc12 71645,C=CCC(CNC(=O)C(CC)N(C)C)C(=O)N(CC)CC1(O)CCC1 71646,c1(C(=O)OCC2CC2)ccccc1NCCCn1cccc1 71647,Cc1cccc(CC(=O)NC2CN(C(C3(O)CCSC3)=O)CC2C)c1Cl 71648,C(=O)(CC1=Cc2ccccc2C1)N1CCC(NC(c2ccc(F)cn2)=O)C(F)C1 71649,C(=O)(CCC(C)(C)C#N)N1C(C(=O)NCC(C#C)OC)CCCC1 71650,c1(OC)cc(O)ccc1NC(C1CSCCN1C(=O)Cc1cc(Br)cs1)=O 71651,C1(CNC(=O)C(C2CCN(C(=O)C3CC3)C2)F)Cc2ccccc2C1 71652,C1(C)(C(N(CCCN(C(C2CCN(C)C2=O)=O)C)C)=O)CCS(=O)(=O)CC1 71653,N1(c2nnc(C(C)(F)F)n2CC2(C)CCCO2)CCNC(=O)C1(C)C 71654,C(=O)(CS(N)(=O)=O)NC(C)CNC(c1ncnn1C1CCOCC1)=O 71655,N1(C(C2CN(C)C2)=O)CCC2CCC12CNC(c1ccoc1Br)=O 71656,N1(C(C(C)O)=O)CC2COCCC2(NC(C2(c3ccccc3Br)CC2)=O)C1 71657,C(=O)(C1=NN(C2CC2)C(=O)CC1)NCCCN(C(C1CCO1)=O)CC 71658,c1(C(CNC(C2(C(=O)OC)CC2)=O)N(C(=O)C(Cl)=CCl)C)ccccc1 71659,CC1CCC=C1C(=O)N(C(C)C(=O)NC1CCC12CCCC2)C 71660,N1(C(CNC(CC)=O)=O)CCC(C(=O)NCC2(C)CC3CC3C2)C(C)(C)C1 71661,C1(NC(=NCCCC)NCC(=O)NCC2CCCO2)CCc2cnn(C(C)C)c2C1 71662,N1(C(C2CC(NC(C(CCOC)OC)=O)C(O)C2)=O)CCOC2(CC2)C1 71663,c1(C(C(=O)NC2CCCC(NC(C(CC)(C)C)=O)C2)O)ccc(F)c(Cl)c1F 71664,CON(C(=O)C1=C(F)CN(C(c2cc(O)ccc2F)=O)CCC1)C1CCC1 71665,C(CCC(=O)NC1(CO)CN(C(=O)C(C=C)OCC)C1)OCC=C 71666,c1(C(C)C)cc(NC(=O)C(=O)NCC2NCCC2C)ns1 71667,N1(C(C(CC)CCOC)=O)CCC2(CC1)CCN(C(c1ccc([N+](=O)[O-])[nH]1)=O)C2 71668,C#Cc1ccnc(C(=O)N(CCCNC(=O)CCn2ccnc2)CCC)c1 71669,C1(N(C(C(C(=C)C)(C)C)=O)C)CCCC2CN(C(c3ccn(C(F)F)n3)=O)CC12 71670,C(C(=O)N=c1cc(C)n(C2CC2)[nH]1)C1N(C(c2ccc(C)cc2C)=O)CCOC1 71671,C(=O)(C(C)N(C(C)COCCOCCOC)C(C)C)OC(C)C 71672,Cc1cc(NC(C2CC(F)(CO)C2)=O)n(-c2ccc(F)cc2)n1 71673,N1(C(C(C)Cc2ccccc2)=O)CC(NC(C2CC(CF)C2)=O)CC(O)C1 71674,CN1CCC(C(=O)N(C)CC2CCCN(C(=O)CC3CCCSC3)C2)CC1 71675,CC(C)CC(C)CC(=O)NC(C)CN(C)C(c1cccc2ncoc12)=O 71676,c1(NC)cc(C(=O)NC2(C)CC(NC(C3CC3Cl)=O)C2)cc(Cl)n1 71677,C1(C)(C(N(CCCC(=O)NC)C)=O)CC(O)CN1C(C1CCN(C)CC1)=O 71678,c1(C(=O)NCC23OCC(NC(COCCCC)=O)(C2)C3)cc(N)ccc1[N+](=O)[O-] 71679,c1(C(N(C2CCN(c3nnc(CC)o3)CC2F)CCC)=O)cc(C)c(C)nc1O 71680,c1(C(=O)NCC=C)cc(F)ncc1NC(c1ncccc1C(F)F)=O 71681,CC1CCCn2c(CC(N3CC(CCNC(=O)CCc4ccoc4)C3)=O)cnc21 71682,N1(C(C(CO)NC(C(C2CCCCC2)C)=O)=O)CCC2CCC(C1)N2 71683,c1(OC)ccc(F)cc1C(C1=CCCCC1)N(C)Cc1ccccc1N1CCCC1 71684,C(C(C)(C)CC(=O)N1CCCC1Cn1cc(CCCN(C)C)nn1)OC 71685,c1(C(=O)NC(CNC(c2ccc(COC)o2)=O)(C)CO)ccncc1OC 71686,Cc1cc(C(=O)NC2CC3CCC2CC3NC(=O)C(O)CC2CC2)cc(C)c1N 71687,c1(C(C(=O)NCCCOCC2CCCN2C(=O)CC2CC2)O)ccc(Cl)nc1 71688,N1(C(C(C=C)(C)CC)=O)CCN(C(c2ccsn2)=O)CC2(CC2)C1 71689,C1(COC)CN(C(=O)Cc2ncoc2C)CCN1C(=O)C1=CCCCC1 71690,c1(-c2n(CCCO)nc(Cc3cccs3)n2)nc2n(c1Cl)CCCC2 71691,c1(OC(C)C(=O)NCC(C)(C)CN(C)C)cccnc1 71692,c1(NCC)cccc(C(=O)N(CCC(C)NC(c2snnc2C)=O)C)c1 71693,C1(C(=O)NCc2ccn(CC)n2)CC(C)(C)CN1C(=O)Cc1cncs1 71694,c1(C(=O)NC(CNC(c2cc(C)no2)=O)CO)oc2ccccc2c1CS(C)=O 71695,S(=O)(=O)(c1ccc(C#N)c(NCC(C)(C)F)c1)N(CCCCC)C 71696,C1(NC(c2occ(C)c2)=O)CCC2(CCN(C(=O)Cc3nc(C)sc3C)CC2)C1 71697,c1(C(C)CC(=O)NC2CC(F)(CNC(=O)Cn3ncnn3)C2)cncc(F)c1 71698,C(=O)(C(C)(C)C(F)(F)F)NC1CC(C)CN(C(=O)CCCN(C)C)C1 71699,C1(C(N2C(C(=O)NCCC3(O)CCC3)(CC)CCC2)=O)CC2C(C1)C2(F)F 71700,C1(CNC(CO)CO)C2(CCC2)C12CCC2 71701,CCCCCC(C)(C)C(=O)N1CCOC(CNC(=O)CC(C)N(C)C)C1 71702,c1(NC(C(=O)Nc2cccc(C3CCC(=O)N3)c2)=O)cc(Cl)n2nccc2n1 71703,C1(NC(CC(COC)C)=O)C2CC3CN(C(C4CCC(C(=O)OCC)C4)=O)C1C3C2 71704,C1(C(=O)NCC(=C)C(F)(F)F)CN(C(c2ccn(C(F)F)n2)=O)CCC1O 71705,C(C(C)(C)OCCOCC(=O)OC(C)(C)C)NC(COCC1CC1)=O 71706,Cc1cc(O)c(C(N2CC(F)CC2C(=O)Nc2cnncc2Cl)=O)cc1Br 71707,c1(OCCC)ccc(S(=O)(=O)NC)cc1C(=O)N(C1CCCCCC1O)C 71708,c1(CC(=O)NCC2CN(C(C3(CC4CC4)CCC3)=O)CCO2)ccc(Cl)c(F)c1 71709,N(C1CCCc2c[nH]nc21)C(CC(CNC(c1cc(CC)nn1C)=O)O)=O 71710,c1(C(C)=O)cc(=NCCC2CCCN(C(C3CCCC3)=O)C2)[nH]cc1[N+](=O)[O-] 71711,C1(CC(=O)NCC2(OC)CCN(C(c3ccc(F)cn3)=O)C2)CC(O)C12CCC2 71712,N1(C2CCN(C(C(C)(C)N3CCCC3)=O)C2)CCN(C(=O)Cc2cccs2)CC1 71713,c1(CC(N2CCCCC(NC(c3nc(C)sc3)=O)C2)=O)ccc2c(c1)CCCO2 71714,N1(C(c2cc(CC)[nH]n2)=O)CCC(C(C)CNC(=O)Cc2cnccc2Cl)CC1 71715,N1(C(C(CC(C)C)ONC(=O)CC2CC3C=CC2C3)=O)CC2(CCOC(=O)N2)C1 71716,c1(CC(N2CC(C(C)NC(c3cccc(=O)o3)=O)OCC2)=O)ccc(O)c(F)c1 71717,CC1(C)CCCC1(N)C(=O)NCc1cn(C2C=CCCC2)nn1 71718,N1(C(c2n(CCC)ncc2)=O)CCCC2CCN(C(c3cnsn3)=O)CC12 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71877,CC1=C(C(=O)NC2CC2NC(C2(C)CC(C)C2)=O)CCC1 71878,N1(C(C2N(Cc3n(C)ncc3Br)C3C(C2)C3)=O)C2CCCC1COC2 71879,C1(NC(C(C(C)C)O)=O)CC2CN(C(c3cc(N)c(Cl)cn3)=O)CC2C1 71880,c1(C(N(C)CCOCCNC(C2CC(C(F)F)C2)=O)=O)ccn2c(O)nnc2c1 71881,Cc1nc(O)ccc1C(=O)NC1CC(C)N(C(=O)CN2CCCC2=O)C1 71882,N1(C(C(C)n2cncn2)=O)CCC2(CCN(C(=O)CN3CCCC3=O)C2)C1 71883,N1(C(C2C(=C)CC2)=O)CCC2(CCC2NC(=O)Cc2ccc(Cl)cc2C)CC1 71884,c1(CCNC(c2n(CCCOC)nnn2)C2(CSC)CC2)nc2c(s1)CCCC2 71885,C1(O)(CNC(=O)CCOCC2CC2)CCCN(C(=O)C(O)c2ccsc2)CC1 71886,O=C1COc2ccc(CC(=O)NNC(=O)Nc3cncc(F)c3)cc2N1 71887,C1(C(N(CC(C)O)CCNC(c2cccc(O)n2)=O)=O)CC2(CCC2)CO1 71888,c1(-c2cccc(NC(c3c(OC(C)C)cccn3)=O)n2)ccc2scnc2c1 71889,CC1(C)CN(C(C2C3CCC23)=O)CCC1NC(=O)CCC1OCCO1 71890,C1(C)(C(=O)NCC(CNC(C2C(C(C)C)CCC2)=O)O)Cc2ccccc2C1 71891,C1(CCC(=O)Nc2c(C)scc2)COC(C)(C)N1C(=O)OCc1ccccc1 71892,N1(C(CCOC)=O)CC2OCC(NC(=O)C(C)(C)Oc3ccc(F)cc3)C2C1 71893,c1(C(N(C)CC2CCCN2C(=O)CN2CC(C)(C)C2)=O)ccc2c(n1)CCCC2 71894,N1(C(CCCCC=C)=O)CCCCCCC1CNC(=O)CCC1CCC(=O)NC1 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71913,N1(C(C23N(C(C4CCN(CC)C4)=O)CCC2C3)=O)CCCC(F)(F)C1 71914,C(C(C)C)(C(O)C(=O)N1CCC(CCNC(C2CCC(=O)N(C)C2)=O)CC1)OC 71915,C1(C)(C(=O)NC2CC(CNC(CC(C=C)(C)O)=O)C2)CC(C(C)C)=NO1 71916,CC1CCCC(NC(=O)C(=O)NC(C)(CNC(c2ccno2)=O)CO)C1C 71917,O=C1CCC(C(=O)N2CC3CC2CN3Cc2c(F)cc(Cl)cc2Cl)=NN1 71918,c1(C(C)=O)nc(C(=O)NCCC2CCN(C(=O)Cn3nnc(=O)[nH]3)C2)cs1 71919,C1(NC(c2nc(OC)oc2)=O)CCCN(C(=O)COC2CCC2)CC1 71920,C12(C(=O)NC(COCC)C)CCC(NC(c3c(C)ccnc3C)=O)(CC1)C2 71921,CC1CS(=O)CCN1C(=O)C(CCN(C)C)NC(=O)C=Cc1cn(C)nn1 71922,C1(CCN(CCOCC#C)C)CCN(C(c2cn(C)nc2-c2ccoc2)=O)CC1 71923,Cc1cc(-c2nc(CCCO)nn2-c2ccccc2C)cnc1O 71924,Cc1cc(C)c(C(=O)N(C)CC=CC(N2CCCC(N(C)C)C2)=O)s1 71925,C1(C(=O)NC(CCC)CC)C2CC3C(C2NC(C2(COC)CCC2)=O)C13 71926,c1(C(C)=O)c(NC(C23CC2CN(C(c2ccc(C#N)s2)=O)C3)=O)cccc1F 71927,C#CC1(C(=O)NC(C(C)C)C2CC2)CN(C(c2ccc(C)cn2)=O)C1 71928,N1(C(C2(NC(=O)CC3CC4(CCC4)C3)C(C)CCC2)=O)CCC2(CCOC2)CC1 71929,C(CCCCN(C)C(C1(CCN(C)C)CC1)=O)NC(C(C)OCCOCC)=O 71930,c1(C(N2CCOCC(CNC(C(C3CC3)OCC)=O)C2)=O)cc(C)cc(C#N)c1 71931,c1(C(N2CCC(CNC(Cc3ccc(C)s3)=O)C2)=O)cc(O)nc(O)n1 71932,C(=O)(CCC(F)(F)C(F)F)N(C)CC1CCCN(C(C2CCC(=O)N2)=O)C1 71933,C1(C(=O)OC)CC(NC(=O)OC)(Oc2ccccc2)C1.C12CCN1OC2=O 71934,C1(C(N(C(c2ccccn2)C)CC)=O)CC2CC(NC(=O)NC3CCCC3)C2C1 71935,C(=O)(C(=O)CCC(C)(C)C)NC1C(CNC(C(CCC)C)=O)CCC1 71936,C1(CC)CCCCC1C(N1CCCC1C1CCN(C(=O)C(=O)NC2CC2)C1)=O 71937,CC(C)C(C)CC(=O)NCc1ncccc1C(=O)NC(c1ccn(C)n1)C 71938,Cc1cc(C(=O)NC2C3CN(C(=O)Cc4cnco4)CC23)nn1CC(F)(F)F 71939,CCCCC(CC(=O)NC1CCC(OC)CC1)NC(c1ccc2cc[nH]c2c1)=O 71940,c1(CC(=O)NCC(C)NC(c2occ(OC)c(=O)c2)=O)noc2ccc(O)cc12 71941,C(=O)(C(C1=CCCCCC1)N1CCCCCCCCCC1)NC(C)(C)C 71942,C1(C(N(CC(=O)N)C(C)C)=O)CCN(C)C1CC.C1(OCC)(CC)CC1 71943,n1(C(C)C)cnc2c(NCCn3ncc(Br)n3)[nH]c(=NCC3C4CCCC34)nc12 71944,CC1OC2(C(=O)NC3CCC(NC(c4cnc(-c5cccs5)[nH]4)=O)CC3)CC1C2 71945,c1(CC(C)C(=O)NC2(C)CN(C(=O)CC(C)N(C)C)C2)ccc(Br)cc1 71946,N#CCCCC(=O)N(C(Cc1cn[nH]c1)C(=O)N1CC(Oc2ccccn2)C1)CC 71947,CC12CCCC(C(N3CCC(c4cn(C5CCCC5O)nn4)C3)=O)(CO1)C2 71948,c1(OCC(C)NCCC(C)C)cccc(Br)c1 71949,CCCC(C(=O)N1CC2CC(NC(c3coc(CC)n3)=O)CC1C2)S(N)(=O)=O 71950,CC(CC(=O)NCC1CCN(C(=O)CC=CCc2ccccc2)C1)CC(F)(F)F 71951,N1(C(c2c(N)nccc2)=O)CC2(CCC(CNC(=O)Cc3cccs3)O2)C1 71952,C1(NC(Cc2c(F)ccc(C)c2)=O)CC12CCC(NC(=O)C(C)CF)CC2 71953,C1(N(C)C)(CC)CCN(C(c2ccc(CNC(C3CC4(CCC4)C3)=O)o2)=O)C1 71954,Cc1ccnc(C)c1C(=O)NC(C)C(C)NC(C1(c2ccccc2Cl)CC1)=O 71955,c1(-c2nc(Cc3c(C)occ3)n(CC(F)F)n2)ccc2ccccc2n1 71956,Cc1cc2cccnc2nc1C(=O)NCCC1CC(NC(c2ccccc2)=O)C1 71957,N1(C(Cc2ncc(C)s2)=O)CC(NC(=O)CS(=O)(=O)C2CC2)C(C2CC2)C1 71958,CC(C)CC(C(=O)NC(C)C(C)NC(=O)CSc1cn[nH]c1)N(C)C 71959,C1(C(=O)NC(C)(C(=O)NCCc2cc[nH]n2)C2CCC2)CCCC(F)C1 71960,c1(CC(=O)NC(CC(=O)NCC2CCC(C)(C)O2)CC2CC2)ccc2c(c1)CC2 71961,C(=O)(C(C(C)(C)C)C1CC1)NC1C(C)CN(C(=O)C(c2ccccc2)N(C)C)C1 71962,c1(C(N2CCC(CCOC)(NC(C(CC=C)C)=O)C2)=O)ccc(C(C)=O)nc1O 71963,C1(NC(C2CCCO2)=O)C2CN(Cc3ccc(OCCO)nc3)CC12 71964,c1(C(N(C)CC2CCN(C(c3cscc3Br)=O)CC2)=O)cc(F)cc(F)c1Cl 71965,C(N=c1[nH]c(=N)[nH]c(=NC(C)Cn2ccnc2C)[nH]1)C1(OC)CCCC(C)(C)C1 71966,C(=O)(CC(C)(C)C(=O)NCC1CCN(C(=O)COCC(C)C)C1)OCC 71967,C1(F)(C(=O)NCC2N(C(c3cccc(O)n3)=O)CC2)C(F)(F)C1(F)F 71968,C(C1=CCCCCC1)(c1ccccc1)N(CC(C1C2CCCC12)=O)C 71969,C1(C(N2C(C(C)(C)NC(C(C)NC(=O)NC)=O)CCC2)=O)CCC2CC2C1 71970,N1(C(C(CCC)(C)O)=O)CC2(CC(NC(=O)Cc3cccc(C#C)c3)CO2)C1 71971,N1(C(C(CC)Oc2ccccc2)=O)CCC2CC1CN2C(c1csc(CO)n1)=O 71972,N1(C(CCCCCSC)=O)CC2CCC(N=c3[nH]ccnc3F)CC2C1 71973,c1(C(=O)NC2(CO)CCN(Cc3n(C(C)C)ncc3)CC2)cccc2cc[nH]c12 71974,CCCCC(CC(=O)Nc1ccc(C(C)C)nc1)NC(=O)CCn1cncn1 71975,c1(C(=O)NC2CC(C)N(C(=O)CC3CSCCO3)CC2)cccc2nn(C)cc12 71976,CC1CN(C(c2cc(Br)co2)=O)CC1CCNC(C1(O)CCC1)=O 71977,N1(C(C2(F)CCN(C(C3=C(C)CCC3)=O)CC2)=O)C2CCC1CC(O)C2 71978,c1(C(N(C2CN(CC3(C(=O)NN4CCOCC4)CC3)CC2F)C)=O)cc(O)ncn1 71979,C1(NC(c2cnn(C(C)C)n2)=O)CCCCCC1C(=O)NCC(c1cnc[nH]1)C 71980,N#Cc1ccc(C(N2CCC23CN(C(=O)Cc2ccc(Cl)cc2F)C3)=O)c(Cl)c1 71981,CC1(C(N2CC(N(C)C)C(CNC(=O)CC3CCS(=O)(=O)C3)C2)=O)CCCC1O 71982,C1(NC(c2cc(C(C)C)n(C)n2)=O)CC2(C1)CC(CNC(=O)C=CCF)C2 71983,C1(NC(Cc2nc(C)sc2)=O)CCOCC1C(=O)NCCc1ccncc1 71984,C1CCCCC1NC(C1C(C(N2CC(=C)C2)=O)C1)=O.C(COC)O 71985,Cc1nc(O)sc1C(=O)NC(c1cn(C)nn1)C(=O)NCC(c1ccccc1)F 71986,C(CN=C(NC(C)CC1CCOCC1)N1CCC(C2CC2)CC1)OC 71987,N1(C(c2cnc3cc(C)nn3c2)=O)CCC2(C1)CN(C(=O)C=C(Cl)Cl)CCO2 71988,Cc1nn(C(F)F)cc1-c1ccc(CNC(C(C)C)C(C)C)cc1 71989,Cc1cc(C(C)C2CC2)nc(SC(=O)C(F)Oc2ccccc2)n1 71990,C1(C(=O)NC(CC)CN(C)C(c2coc(C)c2)=O)COc2cccc(OC)c2C1 71991,C(=O)(C(CCC1CCCO1)N1CCC(Cc2nccn2C)C1)NCCSC 71992,c1(C(N(CC(O)CNC(=O)Cc2ccccc2)C)=O)ccc([N+](=O)[O-])n1C 71993,c1(C(C)C)ncsc1C(=O)NC(C)CN(C)C(c1ccnn1C1CC1(F)F)=O 71994,Cc1ccc(O)c(N(C)Cc2csc(Br)c2Br)n1 71995,N1(C(c2cccc(OC)n2)=O)CC2CCC1C2NC(C1CC(N2CC(O)C2)C1)=O 71996,N1(C(C(CSC)C)=O)CCN(C(=O)CCn2cc[nH]c(=O)c2=O)C2(CC2)C1 71997,FC1(F)C2CCC1CN(CC(=C1CCOCC1)Br)C2 71998,c1(C(N(CCC)CCNC(c2ocnc2C2CC2)=O)=O)c(C)cccc1F 71999,C1(CNC(c2ccoc2)=O)CCCCC1NC(C1CC(O)(C(F)(F)F)C1)=O 72000,N1(C(Cc2cccc(OCC)c2)=O)CCCC(NC(C2(CC(C)C)CC2)=O)C1C 72001,CCC(CC(=O)N1CCC1C(N1CCC(C)(O)C1)=O)SC 72002,C(C(C)C(C)C(=O)NC1C2CC1CN(C(C1CSCCS1)=O)C2)OC 72003,C(=O)(C(C)CCCC(C)C)NC1C(NC(c2c(SC)cccc2)=O)CCC1 72004,C#CCC(O)C(=O)NCC1(C(F)F)CCN(C(C2CC(c3ccccc3)C2)=O)C1 72005,c1(C(=O)NCCCCCCNC(C(F)=CCC)=O)ccc(S(N)(=O)=O)c(N)c1 72006,C#Cc1cccc(OCC(=O)NC2(F)CCN(C(=O)CCCNC(N)=O)CC2)c1 72007,c1(OCC)cc(NC(=O)NCC2(c3oncc3C)CC2)cc(C)c1 72008,C1(NC(CSC)=O)C2CC3CN(C(C4C5CCC(=O)C45)=O)C1C3C2 72009,CN1C(=O)Cc2c(C(=O)NCC(C)(C)NC(=O)C(F)C(F)(F)F)cccc21 72010,C12(C(N3CC(C)(NC(c4cc(Br)n[nH]4)=O)C3)=O)CCC(C1)S(=O)(=O)CC2 72011,c1(C(=O)NC(CCOC)CNC(c2cnc(C(C)C)s2)=O)cncc(C)c1C 72012,c1(-n2c(C3CC3(C)C)nc(C(CCC)C)n2)ccc(F)cc1C(F)(F)F 72013,Cc1cccnc1CCC(N1CC2CC2(NC(=O)CSCCC#N)C1)=O 72014,C(=O)(C1=CCCSC1)N1C(CCCNC(CNS(CCOCC)(=O)=O)=O)CCC1 72015,C1(CC(=O)NCCC2CC(NC(=O)C=CC3CCCC3)C2)CC(F)(F)C1 72016,CC1(C)CCCC(C(N2CCC(CO)(NC(C3CC(F)(F)C3)=O)C2)=O)C1 72017,c1(SCC)cc(C(=O)NC2(C(F)F)CC(NC(=O)C(C)CSC)C2)ccn1 72018,c1(CCCNC2(c3n(C(CC)C)nnn3)CCCC2)ncccc1C.C(CO)S 72019,N1(C(C(CCSC)O)=O)CC2CC1CCC2NC(c1cc(C)c(F)c(C)c1)=O 72020,N1(C(CCC2CC(NC(C3C(C)CC(=O)NC3)=O)C2)=O)CCCN(C)CC1C 72021,N1(C(c2n(CC=C)ccc2)=O)CCC(C)(C)C(CNC(c2ccsc2C)=O)C1 72022,N1(C(c2cc(OC)nn2C)=O)CCC(CO)(NC(c2snnc2C)=O)CC1 72023,c1(NCc2cn(C3C(NC(CC)=O)COC3)nn2)ncccc1C(=O)O 72024,N1(C(C(C)(C)CCl)=O)C2CCCC1CN(C(C1CCc3ccoc3C1)=O)C2 72025,c1(C(=O)NCCCCC(C)NC(c2c(CC)non2)=O)c(O)cc(Cl)cc1F 72026,C12(NC(c3cc(CC)n(CC)n3)=O)CCC1CN(C(C1CCOC(=O)CC1)=O)C2 72027,c1(NCC)cccnc1C(=O)N(CC(C)CNC(=O)C(c1cccc(Cl)c1)C)C 72028,C(=O)(CN=S(C)(C)=O)NC1(C)CC(NC(C2CC2C2CCCO2)=O)C1 72029,CC1(C)C(CNC(=O)C(O)C2CC2)CCN1C(=O)CCCN1CCCC1 72030,C(=O)(CCCCC#N)N1CCCC(CC(=O)NCCn2c(C)nnc2O)C1 72031,c1(CC(=O)OCC)cccc2c1CCN(Cc1n[nH]c3c1CCC3C)C2 72032,c1(C(=O)NCCCN(C(=O)CC2(C(F)(F)F)CC2)CCO)n[nH]c(O)n1 72033,c1(C(N2CC(CNC(c3c(O)cccc3O)=O)OCC2)=O)ccc(Br)cc1F 72034,CC(C)(C)C(O)C(C(=O)NCC(c1ccco1)O)C1CCCC1 72035,S(=O)(=O)(c1cccc(Cl)c1)NCC(N1CCC(N(C)C(c2cccs2)=O)C1)=O 72036,C12(C(=O)NC3CCC(N(C(=O)CCNC(=O)CO)C)CC3)CC1CCC2(F)F 72037,C(=O)(C(C)C(C)NC1(CC(=O)C2CC2)CC1)OC.C12CCC1CNC2=O.C1CN1 72038,N1(C(C2N(C(C)C)C(=O)CC2)=O)CC(NC(C2C(C)(C)OC2(C)C)=O)CCC1C 72039,C1(CNC(C=CC(C)(C)C)=O)CC2COCC2N1C(C1(F)CC2(CCC2)C1)=O 72040,N1(C(C(CC#C)CC#C)=O)CCC2C(C1)NC(=O)CN2C(=O)CCCC(C)CC 72041,c1(NCC2(C#N)CC2)cnc(F)cc1C(=O)Nc1cc(Br)cc(I)c1 72042,C1(CNC(=O)C2=CCCC2)CCC12CCN(C(c1cnc3ccsc3c1)=O)CC2 72043,N1(C(C(CC)F)=O)CC2CC1CN2C(c1ncsc1Br)=O 72044,CCC(C)(C(=O)N1CC(CNC(=O)CO)C1)C(N)=O.CCCC(C)N(CCC(=O)O)C 72045,N1(CCO)CCC(N(C2CCN(C(C)C)C2=O)C(=O)C(F)=C2CCCC2)CC1C 72046,C1(N(C(CN(C(C=CCOC)=O)CC(C)C)=O)CC)CCC2(CCC2)CC1 72047,C1(NC(c2ccc(O)cn2)=O)C=CCN(C(c2ccncc2C2CC2)=O)C1 72048,N1(C(C(CC=CC)C)=O)CC2CC1CC2CNC(=O)CCNC(=O)CO 72049,N1(C(C(COC)NC(=O)C(C)C#N)=O)CCC(F)(CF)CC1 72050,N1(S(CC2CCC(N(C)C(=O)OC(C)(C)C)C2)(=O)=O)CCOC(CC2CC2)C1 72051,N1(C(CC(=C=C)C)=O)CC2(CCCN(C(=O)COC(=O)Nc3ccncc3)C2)C1 72052,C1(C#N)(NC(c2cc(C(=O)OCC)no2)=O)CCCCCC1 72053,c1(C(N(CC(CC)NC(C2CSCCS2)=O)C)=O)cc(C)c(C)o1 72054,C1(C(=O)NC2(CC)CCCC2)CN(C(C2CC23CCCC3)=O)CC1(F)F 72055,c1(C(=O)NCCc2ccc(CNC(C=CS(C)=O)=O)cc2)nc2cnccc2s1 72056,c1(C(=O)NC2C3CN(C(c4n[nH]c(C)c4C)=O)CC2C3)cn2c(n1)CCC(C)C2 72057,c1(C(=O)NCCC(C)N(C)C(C2CCCC3CC23)=O)ccc(-c2ncc[nH]2)nc1 72058,N1(C(=O)CC2CCN2C(=O)CCc2ccco2)C2CCC1COC2 72059,C1(C(=O)NC2C3(CC(NC(c4ccnnc4)=O)C3)C2)CC12CCSCC2 72060,O=C(C1CCCc2nccn21)NC1CC1C1CCN(C(=O)C=C2CCC2)CC1 72061,c1(OC(C)C)nc(F)ccc1-c1cc(NC(=O)C(C)(C)O)ccn1 72062,Cc1scc(C(=O)NCC2CCCC2NC(c2ccnc(SC3CC3)c2)=O)c1C 72063,c1(C(=O)NCC2N(S(CCCC)(=O)=O)CCCC2)cc(Cl)cc(OC)c1O 72064,N1(C(CC2C(C)=NOC2=O)=O)CC(NC(c2onc(C)c2C)=O)CC1(C)C 72065,Cn1cc([N+](=O)[O-])c(C(=O)NC2CC(NC(c3coc(Cl)c3)=O)C2)n1 72066,Cc1c(C(N2CCC(CNCc3ccc4cc[nH]c4c3)CC2)=O)cc(F)cc1Cl 72067,N1(C(c2cc(C(C)=O)[nH]n2)=O)CC(n2cc(CN3CCCC3)nn2)CCC1(C)C 72068,c1(NC(CCN(C(C2C(OC)(OC)CC2)=O)C)=O)ccncc1C(C)C 72069,N1(C(C(C)CCO)=O)CC(C2CCCN(C(=O)C(C)(O)C3CC3)C2)C1 72070,N1(CC(=O)NC(c2ccc(Cl)cc2)C(=O)OC)CCC(C(=O)N(C)C)CC1 72071,c1(CN2C(C(=O)NC3CCC(C(N)=O)C3)COCC2)c(Cl)ccc(F)c1F 72072,CC(CNC(=O)CCC(N)=O)C(F)C(=O)NCCCC(C)(C)C 72073,C1(C2(O)CCN(C(=O)CCC(N)=O)CC2)(NC(c2ncc(C)nc2)=O)CC1 72074,N1(C(C=CC(F)=CCC)=O)CCC(C(=O)OC)CC1C(=O)OCC 72075,CCS(=O)(=O)CC(=O)NCC1(F)CC(NC(=O)CC2CCC2(C)C)C1 72076,Cc1cc(CNC(=O)CC(O)CNC(C2CCOC2)=O)sc1C 72077,c1(CC(N2CCC(C)(CNC(C3C(C)C3C)=O)C2)=O)ccc(F)c(F)c1 72078,CC(C)C(O)CC(=O)N(C(C)CCNC(=O)Cc1ccc(Cl)cc1F)C 72079,c1(C(=O)NC2C(NC(CSC)=O)CCCC2)cc(Cl)cc(C)c1O 72080,C1(NC(c2sc(CC)c(C)c2)=O)CN(C(C2(C)CC(C)C2)=O)Cc2ccnn2C1 72081,CC1(CN(C(C2(c3ccncc3)CC2)=O)C2CC2)CCN(C(=O)C(N)=O)C1 72082,c1(C(=O)NC(CC)CNC(C2C=CCC2)=O)csc2ccc(Br)cc12 72083,CCC(O)C(F)(F)C(=O)N1CC2(CNC(c3cc(C)on3)=O)CC1CO2 72084,C1(NC(=O)C=Cc2ccccc2)CN(C(=O)C(O)CC2CC2)CCC1C(F)(F)F 72085,c1(NCC(C)N(CC)CC)nc(N2CCOC(C)(c3ccccc3)C2)cc(C)n1 72086,C1(NC(C2(c3nc(Cl)cc(OCC)n3)CCC2)=O)CC2CCCCN2C1 72087,C(CCCCCNC(C12CC(NC(C3CC3(C)C(C)C)=O)(C1)C2)=O)OC 72088,C1(COCC(=O)NC2C(CNC(=O)COCC3CCC3)CC2)CCCOC1 72089,N1(C(c2c(C)nc(F)cc2)=O)CCC2(CC1)CCN2S(=O)(=O)c1ccc(Cl)cc1 72090,n1(CC(C)O)nc(COc2cnn(C)c2)nc1-c1ccc(=O)oc1 72091,C(C(CC(C)C)C(=O)N1CCC(CNC(=O)C(C)CO)(COC)CC1)OC 72092,C(C)(CN=C(NCC(=O)NC1(C)CC1)NC1CCC1)OC 72093,C#CC1(NC(=O)NCC2CN(C)C(=O)N2)CC(=O)C1 72094,c1(N(S(CC)(=O)=O)C)nnc(N2CCOC(c3nccs3)C2)n1CC1CC1 72095,N#CC1CN(C(c2ncc(F)cc2F)=O)CCN1C(c1sccc1Br)=O 72096,CC(C)C(C(=O)NCC(C)(Cn1cccn1)NC(=O)C=Cc1ccc[nH]1)NS(C)(=O)=O 72097,C1(C(=O)NOCCC2CC2)(CC)CN(C(=O)C(CC)OC)C1 72098,C(=O)(CCCCC#N)NCc1cccc(C(N(C(C)C(=O)NC)CC)=O)n1 72099,Cc1cc(C(=O)N(C(C)CNC(=O)C(c2cccc(Cl)c2)C)C)oc1C 72100,C#CC1(C(=O)N(C2CCOC(C)(C)C2)C)CCN(C(=O)COc2ccsn2)CC1 72101,N1(C(c2c(NC)cncc2)=O)CCC2(COC(CNC(=O)C(C)(C)CO)C2)C1 72102,c1(CNC(=NCC23CC(C)(OC2)C3)NCC2CCCCC2)cc(Cl)cnc1F 72103,C1(C(=O)NCC(C(C)O)C)N(C(=O)Cn2cncn2)CCC1(C)C 72104,C1(C(=O)NCC(CNC(C2N(C(=O)NC)CCC2)=O)(C)C)C2CNC(=O)C12 72105,C1(C(N(C)CC2(NC(c3ccc(N)cn3)=O)CC2)=O)CCC(F)(F)CO1 72106,C#Cc1ccc(C(N2CCC(C)(C)C2CNC(C2(N(C)C)CCCC2)=O)=O)cn1 72107,c1(C(N2CCC(C)(C(=O)NCc3ccccc3)C2)=O)cc([N+](=O)[O-])c(F)cc1Br 72108,CC(C(=O)NC1CCN(C(=O)CN2CCOCC2)CC1)C1OCCc2sccc21 72109,CC1CC(N=c2[nH]c(=NCc3cc(Cl)ccc3N(C)C)[nH]c3cc[nH]c23)CC(C)N1 72110,CCCCCC(=O)N(C1CCCC(NC(C2(COC)C=CCC2)=O)C1)C 72111,c1(C(=O)NC(C(C)C)CNC(=O)CC2(C)CC2)ccccc1-c1ccccc1 72112,c1(C(=O)NCC(=C)CCNC(C2(S(C)(=O)=O)CC2)=O)cc(Cl)ccc1Cl 72113,c1(C(=O)NCC2C(C)(C)CCCN2C(=O)CS(N)(=O)=O)ccc2nc(O)[nH]c2c1 72114,N1(C(C(COCC)O)=O)CCC(C)(CNC(=O)C(c2cccc(C(N)=O)c2)=O)C1 72115,c1(C(N(C(C)(C(N2CCCC(F)C2)=O)C2CC2)C)=O)ccc(O)cn1 72116,c1(NC(C(Cc2cnc[nH]2)NC(C(CC)C)=O)=O)ccc2c(c1)OC(F)(F)O2 72117,CC(=O)CCCCC(=O)N1CC(C(=O)NCC2CCCC(=O)N2)CC1(C)C 72118,c1(CN2CCCC(C(C)NC(=O)COC3CCOC3)C2)ccc(F)cc1Br 72119,C1(CNC(c2cc(SC)cc(Cl)c2)=O)CN(C(C2COCCO2)=O)CCC1(C)C 72120,Cc1cn2c(n1)CCC(C(=O)NC1CC3CC1N(C(=O)CC1(C)OCCO1)C3)C2 72121,c1(C(N2CCN(C(c3c(SC)nccc3)=O)C3C2C3)=O)cc2cc(F)ccc2[nH]1 72122,C12(C(=O)NCCOCCN(C)C(c3ccc(CO)s3)=O)CCOC1CCOC2 72123,C(C(=O)NC12CC(C1)N(C(c1ccc(C#N)s1)=O)C2)(C(C)C)n1ncc(C)c1 72124,c1(C(=O)NCC2CCC(NC(C3CCNC3=O)=O)C2)cc2cc(F)ccc2s1 72125,Cc1nsc(NC(C2CC(F)CN2Cc2c(Cl)cccc2Br)=O)c1C#N 72126,C(=O)(C(C)(C)C(C)(F)F)NC(C)CCNC(C1CCC2CC2CC1)=O 72127,C1(OC)CN(C(=NCCCN2CCOC2=O)NC2CCC2)CC1O 72128,Cc1ccc(C(=O)NCCC2CCCN2C(=O)CC2CC23CC3)cc1S(C)(=O)=O 72129,C1(CNC(C2(CNC(CC3C(C)=NNC3=O)=O)CCCC2)=O)OCCCC1(C)C 72130,C#CCC(C)(C(=O)N1CCC(C(=O)OC)O1)NC(=O)C(CC)CC=C 72131,C(CCC)(C(=O)Nc1cccc(CNCCc2ocnc2CC)c1)=CCC 72132,CC12CC(CCO1)N(C(C1CC3(CCN1C(=O)C(N)=O)CC3)=O)C2 72133,C=CCC(CC)C(=O)N1CC2CC(C1)N2C(C1C=CCS1)=O 72134,C#CC1CN(C(=O)C(N2CCC(C(C)COC)CC2)=O)CCN1 72135,C1(NC(c2c(C)coc2)=O)CC(C)CN(C(=O)COC2CCC2)C1 72136,C12(NC(c3nc(C)sc3C)=O)CCC(CN(C(c3ccoc3C(F)(F)F)=O)C1)C2 72137,N1(C(C(CCSC)O)=O)CC2(CCC2NC(=O)Cn2cnnn2)C1 72138,CC1CC(C(=O)NCCOC2CCN(C(=O)CCc3cnn(C)n3)CC2)C1(C)C 72139,c1(C(N2C3(CN(C(CCCCC)=O)C3)CC2)=O)cn2c(n1)C(=O)N(C)CC2 72140,c1(C(=O)NC(C)CCCCNC(=O)C=Cc2ccccn2)ccc2c(c1)CCC2 72141,N1(CC)CCC(C(=O)NC2(C(=O)NC3COCC3CN(C)C)CSC2)C1 72142,C1(=O)C(CN=[N+]=[N-])N1.C(=O)(C(CC)n1cncn1)NCCN(CCC)C(C)C 72143,C1(OC)CC2(C1)CC(C(=O)NC1CNC(=O)CN1C(=O)COC(C)(C)C)C2 72144,C=C(Cl)CCC(=O)N1CCOC(CN(C)C(c2ccc(C(F)(F)F)[nH]2)=O)C1 72145,C1(NC(CCCC#C)=O)CS(=O)(=O)C12CCN(C(=O)C(C)CS(C)(=O)=O)CC2 72146,c1(C(=O)NCC2(O)CN(C(Cc3ccn(CC)n3)=O)C2)cc(C)oc1C(F)(F)F 72147,C1(CC)CCOCCN1C(c1ccc(C#N)s1)C(=O)NC(C)C(=O)OC 72148,C#Cc1cncc(C(=O)NC2COCCC2C(=O)NCCc2cncs2)c1 72149,n1(C(C)C)c(O)nc(N2CCC(NC(c3cc(Cl)ccc3F)=O)CC2C)cc1=O 72150,c1(C(=O)NC(C2CCN(C(CC=C)=O)C2)C)ccc(F)cn1 72151,C1(C(=O)NCCCC(C)NC(C=C(COC)C)=O)CCC(=O)N(C(C)C)C1 72152,C=C(Cl)C(C)(C)C(=O)N1CCC(NC(=O)C(C)C(=O)N2CCOCC2)C(O)C1 72153,CC1CCC(C(=O)NCC(C2CCCC2)NC(c2cc[nH]n2)=O)CC1 72154,[SH](=O)(=O)c1cccc(F)c1.C(CCC(=O)NC(C)(C)CNC(=O)CNC)OCC 72155,N1(C(C(CC#CC)NC(=O)OC(C)(C)C)=O)CCS(=O)(=O)C(CO)C1 72156,C=CCCC(C(=O)N(CCC)CCC)NC(=O)CC(C)C(F)F 72157,C(=O)(C1=C(C)Oc2ccccc2C1)N1CC(NC(CCC#CC)=O)C(OC)C1 72158,C(=O)(CS(=O)(=O)Cc1ccccn1)NCC(N(C)C(C1CC(O)C1)=O)C1CC1 72159,c1(NC(=O)NCCCNC(C2CCCN(C(C(C)C)=O)C2)=O)cc(N)c(F)cn1 72160,c1(C2(C(N3CC(CNC(C45COCC4C5)=O)C(O)C3)=O)CC2)ncccc1F 72161,C(=O)(CC(C)(C)N(C(=O)CCn1ccnc1)C)N(CCN(CC=C)C)CC 72162,C(=O)(C1=CCCCC1)NC(CSCC)C(=O)NCc1cnc[nH]1 72163,Cc1nc(C2CC2)sc1CC(=O)NC1CCCC1NC(=O)CN1CCCC1 72164,N1(C(c2c(Br)ccc(C)n2)=O)CCC2(CCN(C(C3CC3C3CC3)=O)CC2)C1 72165,C(=O)(C(C)C(F)(F)F)N1CC(N2CCN(C(c3c(OC)cncc3)=O)CC2)C1 72166,C1(NC(c2cc(CC)nnc2C)=O)CCN(Cc2nnc(COC)s2)CC1(C)C 72167,C(CCNC(=O)CCSc1nccn1C)(C(C)C)NC(c1ccc(CCC)[nH]1)=O 72168,c1(Nc2cc(NCC34CCCCC3NCC4)nc(C)n2)cc2cc(C)ccc2[nH]1 72169,c1(CCC)c(C(N2CC(NC(=O)COCCOCC)CC2CO)=O)nnn1C 72170,C1(C(=O)OC)(NC(=O)CCc2cccnc2Br)CCN(C(=O)OC(C)(C)C)C1 72171,C1(C(=O)NC(CC(=O)NC)(C)C)CC2(CCC2)CN1C(=O)C(C)N(C)C 72172,C12(C(N(CCC=C)CC)=O)COCC1CN(C(c1cc(OC)n[nH]1)=O)C2 72173,c1(C(=O)NCC2(F)CC(NC(COCC(=C)C)=O)C2)cccn(C2CCC2)c1=O 72174,Cc1cc(C(=O)NC2CC(NC(C3CC3C3CC3)=O)C2)cnc1C(F)F 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72192,C1(NC(c2ccn(C(F)F)n2)=O)CCN(C(c2ncc(Cl)s2)=O)CC1CO 72193,C1(C(C)NC(C2CCC3CC23)=O)CN(C(c2csc(C(C)(C)C)n2)=O)CCO1 72194,CC1CC(=O)NC1C(=O)NCC1CCCN(c2ncc(Br)cn2)C1 72195,Cn1cc(Cl)c(CC(=O)NCc2cccc(NC(C34COCC(C3)C4)=O)c2)n1 72196,N1(C(=O)OC)CCCC(C(N2CCC(OCC(c3ccncc3Cl)=O)CC2)=O)C1 72197,CC#CCCCC(=O)NCCCOCCC(=O)NC1(CO)CCS(=O)(=O)C1 72198,c1(C(=O)NC2C(CNC(CNC(=O)NC)=O)C2)coc(C#Cc2ccccc2)c1 72199,Cc1ccn(C)c1C(=O)NCC(C)CNC(C1(c2ccccc2)CC1Br)=O 72200,c1(NC)ccc(C(=O)NC2CC2NC(c2cc(C(O)C(F)(F)F)ccn2)=O)nc1 72201,CC1CC(C(=O)NCC2CCN(C(c3cc(F)ccc3O)=O)C2(C)C)=NO1 72202,N1(C(Cc2n(C)cnn2)=O)CCN(C(CNC2CCC2)=O)CC1 72203,Cc1c(Br)cnc(O)c1C(=O)NCCCCCNC(C1CCCC(F)C1)=O 72204,O=NN1CCCC1C(=O)NC1C=CCN(C(c2ccc(-c3cn[nH]c3)cn2)=O)C1 72205,Cc1noc(C)c1C(C)(C)C(=O)NCC1(O)CCN(C(=O)COC(C)C)C1 72206,n1(CC)cc(C(=O)NCC(O)CN(C(=O)CCn2ccnc2)C)c(C(C)(C)C)n1 72207,N1(C(c2c(CC)nns2)=O)CCOCC(F)(CNC(=O)CC2CCNC(=O)C2)C1 72208,N1(C(C2CC(=O)NC2)=O)CC2CCC1C(CNC(c1n[nH]c3c1CCOC3)=O)C2 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72228,c1(C(N(C(C)CCNC(c2cnc(S)n2C)=O)C)=O)c(Cl)nc2ccccn12 72229,N1(C(C(C2CC(F)(F)C2)OC)=O)CCCC2(NC(c3cnsc3C)=O)CC2C1 72230,CCC(F)(F)C(=O)NC1C=CC(CC(=O)NCc2ccc(OC)nc2)C1 72231,Cc1ccnc(C(F)(F)C(=O)NCC(C)(C)NC(=O)CC(C)N2CCCC2=O)c1 72232,C1(CC(=O)NCCCNC(C2C(C)(C(F)F)C2)=O)CCSCC1 72233,N1(C(c2ccc(C)cc2)=O)CC(C(=O)N(C2CC2)CC2CC2)CC(C)(C)C1 72234,CN1CCN(C(C2(F)CCCOC2)=O)c2cnccc21 72235,C1(NC(c2ncccn2)=O)CCN(C(=O)CC23CCC(CC2)CC3)CC1F 72236,C1(CNC(c2n(CCCC)nnn2)(C)CSC)CCCC12CCOCC2 72237,Cc1c(Br)csc1C(=O)NC1CN(C(=O)C(O)CN(C)C)CC1O 72238,c1(CC)cc(C(=O)NCC2(C)CC(OC)CN2C(=O)CC2(OC)CC2)cc(C)c1 72239,c1(OC)c(C)cnc(C(c2nnnn2C)NC(c2cncc(Br)c2)C2CC2)c1C 72240,c1(C(=O)NCC2CCN2C(=O)CC2CC=CCC2)cc2c(C3CC3)cccc2[nH]1 72241,C=CCCCC(C(=O)NCCC(F)(F)Cl)NC(C1CNC(=O)N1)=O 72242,C(=O)(C(CC(C)C)NC(C1CC(O)C1)=O)NC(COC)CCO 72243,CCCCCCC(CC)C(=O)N1CCCCNC(=O)CC1 72244,c1(C(N2CC(NC(=O)COCc3ccccn3)C2)=O)ccnnc1S 72245,CC(=O)CCCC(=O)NCC(O)CCNC(=O)CSCc1ccc(C)cc1 72246,c1(C(=O)NCC(CNC(CC(CC)C2CCC2)=O)O)c[nH]nc1S(N)(=O)=O 72247,C(N=c1ccnc(NC2CS(=O)(=O)CC2C)[nH]1)c1cc(SC)ncc1 72248,c1(NC(C)C(N2CCCCC2CNC(c2ncncc2F)=O)=O)ccc(Cl)cc1 72249,C1(C(=O)NCCN(CC)CC)CCC(CNC(C2CC2C(C)(C)O)=O)O1 72250,C1(C(C)C)CCC(C)CC1CN(C(C(=O)Nc1cc(-c2ccccc2)on1)=O)C 72251,Cc1cc(C(N2CCC3C(C2)CN3C(=O)CN2CCC2C)=O)cc(C)c1C 72252,C1(C)(OC)CC(NC(=O)N(C(C)C(C)(C)C)C(c2csnc2C)=O)C1 72253,N1(C(C2(C)CC(OC)(OC)C2)=O)CC(NC(=O)CCC2CCCO2)C2(CC2)C1 72254,N1(C(C(C(C)C)C#N)=O)CCCC2(CCN(C(c3cnn(C(C)C)c3F)=O)C2)C1 72255,c1(C(=O)NCC(C2CCC2)Nc2nccc(C3CC3)n2)ccc2ocnc2c1 72256,C(=O)(CC(F)(F)C(C)(F)F)N1CCCC(C)(CNC(C=CCCC)=O)C1 72257,C1(NC(c2cc(C)n(CC)c2C)=O)CCC2(CC1)CC(NC(=O)CC(C)(C)O)C2 72258,N1(C(C(C)CF)=O)CC2(CCCCN(C(=O)C(C)S(N)(=O)=O)C2)C1 72259,N1(C(c2cnn(CC)c2C)=O)CC(CNC(=O)CC(F)(F)Cl)CC12CCC2 72260,Cn1nccc1CC1CCN(C(c2cc(C(C)F)on2)C(=O)NC2CCOC2)C1 72261,CCC(C)C(=O)NC1CC(O)C1CC(=O)NC(CC)CO 72262,N1(C(C)=O)CCC2(CC1)CN(CC1CCC(C(F)C(=O)O)CC1)CCO2 72263,c1(SC)ncc(N)c(C(=O)N(CCNC(=O)CCc2nc[nH]n2)C2CC2)n1 72264,C1(NC(C(C)O)=O)CN(C(=O)CN2CCC(N(C)C)CC2)CC2(CC2)C1 72265,N1(C(c2ccc(OC)c(Br)c2)=O)CC(NC(C)=O)C(C2CC2)C1 72266,N1(C(=O)NC2CCc3ncccc3C2)CCS(=O)(=O)c2ncc(Br)cc21 72267,C1(n2cc(CCCCC)nn2)CCC(C(N2CCC(n3cnnn3)C2)=O)CC1 72268,C(=O)(C(C)(CC)CCC)N(CC(=O)NC1CC(C(=O)OCC)C1)CC#C 72269,C1(C(=O)NCC2(COC)CCOC2)CC12CCN(C(=O)C(C)=CC(C)(C)C)CC2 72270,n1(CCC(=O)NC2CN(C(C3(C4CCCO4)CC3)=O)C2)c(=O)oc2cc(Cl)ccc12 72271,N1(C(c2c(C)nn(C)c2)=O)CC2(CC(C(=O)NCC3(CN(C)C)CCC3)CO2)C1 72272,C1(NC(C(C)=C2CCCC2)=O)CC2CCC(C1C)N2C(c1cc2cscc2s1)=O 72273,C12(C(=O)NC3CC(CC(=O)OC)C3)CCCC1CCN2C(C1CCOCC1(C)C)=O 72274,c1(OC)ccc(C(=O)NC2CCCC2CNC(C)=O)c(NC(=O)C(C)(C)CF)c1 72275,C1(CC=C)(NC(=O)CCSC(F)(F)F)CCN(C(c2cc(CC)nn2C)=O)CC1 72276,c1(C(=O)NC2(C)CCN(C(c3c(C)cc(Cl)cc3)=O)C2)cnc2c(c1)nnn2C 72277,c1(OC)cncnc1C(=O)NCC(c1ccc(C)cc1)NC(=O)CN(C)C(C)=O 72278,Cc1ccc(OCCC(=O)NC2CN(C(=O)CC3CCC(C)(C)CO3)C2)c(Cl)c1 72279,C1(C2CCN(C(=O)COCCN(C)C)C2)(NC(CCCC)=O)CC1 72280,CCC(CCCC(F)(F)F)NC(=O)C(=O)NC1CCS(=O)(=O)CC1 72281,c1(OC)ccc(CN(C)C)cc1C1CC1.C12(CC1)CC(=O)NCC1CC1NC2=O 72282,C(=O)(C1=CCC(NC(=O)CC2CCCC(=O)C2)C1)Nc1cccc(C(C)=O)c1 72283,CC(C)(F)C(=O)NC1CCCC1CNC(c1cn(CCF)nn1)=O 72284,c1(-n2cc(CCC3N(C(CC)=O)CCC3)nn2)ccc(F)cc1Br 72285,Cc1ccc(NC(c2n[nH]cc2NS(=O)(=O)C(F)(F)F)=O)c(C)c1 72286,C(C(=O)NCCC(O)CNC(=O)CCCN(C)C)(C(C)C)(C(C)C)NC(C)=O 72287,C=CCCCCCCCCC(=O)N1CCN(C(=O)C(O)C=C)C2CCCC12 72288,Cc1cc(=NC2CCC(N3CCOCC3)C2)[nH]c(=NCC2COC(C)(C)C2)[nH]1 72289,CC(C)C(CC(=O)NC1(CCNC(=O)CCc2ncc[nH]2)CC1)C(C)C 72290,C(c1cccc(Cl)c1Cl)=CCN1CCCC(C(=O)OCC)C1c1nn[nH]n1 72291,C1(CNC(C(C(C)C)OC)=O)CCN(C(c2ccc(Cl)c(O)c2)=O)C12CC2 72292,CC1CN(C(C)C(=O)Nc2ccccc2C(N)=O)CCC1O 72293,c1(C(=O)NCC2CN(C(CCCC)=O)C(C)(C)C2)cc(C)cc([N+](=O)[O-])c1N 72294,c1(C(=O)NCC2(c3ccon3)CC2)cccc(N(C)C)n1.C(C1C(=O)N1)OC 72295,c1(C(N2CCN(c3ccnnc3)CC2)C(=O)NC(CC)C)cc(C)oc1C 72296,c1(C(N(C)CC2CCN(C(c3cc(CS(C)(=O)=O)on3)=O)C2)=O)cccc(F)c1 72297,c1(C(=O)NC(C2CN(C(CCCOCC)=O)C2)C)cncc(C)c1C 72298,C1(OC)CC2(C1)CN(C(=O)Nc1nscc1SC)C2 72299,Cc1cccc(NC(=O)Nc2ccc(-n3ccnc3C)nc2)c1C 72300,C(CCCCCN=c1[nH]c(Cl)nc2c1SCC2)N(C(=O)CCCS(C)(=O)=O)C 72301,C1(CC(=O)NCCN(C(c2ccc(OC)nc2F)=O)C)CCC2(CC1)CCC2O 72302,CCCC(C(O)C(=O)N1CCCC1c1nc[nH]n1)NC(c1csc(C)c1)=O 72303,C1(C(=O)NC2(C(=O)NCCC(C=C)(C)C)CCCC2)CC(=O)NC(=O)C1 72304,C12CCCC(C1)CNC2=O.CCC(C(=O)N1CC(N(C)C)C1)N(CC)CC 72305,N1(C(CCc2ncn(C)c2)=O)CC2(C1)CN(C(=O)C(O)CCc1ccc[nH]1)C2 72306,c1(OC)ccc([N+](=O)[O-])c(N2CC(NC(=O)C(C)CO)CC3(CC3)C2)c1F 72307,C(Br)(C(=O)N(CC(O)CN(C(=O)C(=O)NC1CC1)C)C)=C(C)C 72308,C(CCCOC)(C(=O)N1CC(CO)CC1(C)C)NC(c1c(C)cc(CC)o1)=O 72309,N1(C(C(C)OCCC(C)C)=O)CCCC1C=CC(N1CC(O)(CCO)C1)=O 72310,N1(C(C(C)Cc2ccccn2)=O)CCN(CCNC(=O)CC2CCCCC2)CC1 72311,n1(CCC(=O)NCCC(C(C)C)NC(C(C)SCCCC)=O)cnc(C)cc1=O 72312,c1(C(=O)NCC2CCN(C(C3(CF)CC3(F)F)=O)C2)ccc(-n2cncn2)cc1 72313,C12(C(=O)NCCCN(C(C(C3CCC3)OC)=O)C3CC3)CCC(=O)N1CCS2 72314,c1(OC)ccc(C(=O)NCC(CNC(C2CC(F)(F)C2)=O)OC)c(C)n1 72315,c1(C(N2CC(NC(C3(c4cccs4)CC3)=O)C(F)C2)=O)cccc2c1OCO2 72316,C(CCCCC(=O)N1CCC(c2cnco2)C1)NC(c1c(C)c[nH]n1)=O 72317,Cc1ccc(C(=O)NCC(C2CCC2)NC(=O)CN2CCN(C)CC2)cc1 72318,CC1(CNC(=O)C(c2cc(F)ccc2F)=O)CCCN(C(C2CC(=O)N2)=O)C1 72319,N1(C(c2cc(CCC)on2)=O)CCN(C)C(C(=O)OCC)C1 72320,c1(CNC(c2c(C)con2)=O)ccc2c(c1)CCC2NC(=O)C(O)CCC(C)C 72321,C(=O)(C(C)CC(C)(F)F)N1CCC(N(C(=O)Cn2nc(C)n(C)c2=O)CC)CC1 72322,C1(CC(=O)NC2CC(NC(c3cccc(C(N)=O)n3)=O)C2)CC(O)C12CCC2 72323,c1(CN(C(=O)NC(C)CCc2cn[nH]c2)C2CC2)nn(C)cc1Br 72324,c1(C(N2CCCC(CCC=C)C2)=O)coc2c1CN(C(=O)CC1CCCN1C)C2 72325,c1(CNC(C(=O)NCC(CC)Oc2cccc(C)c2)=O)ncccc1C 72326,Cc1c(C(=O)N(C)CCNC(C2(C(=O)OC(C)(C)C)CCC2)=O)nnn1C 72327,C(=O)(C(O)CC(C)(C)C)NC(CCCNC(c1ccc(SCC)nc1)=O)(C)C 72328,C1(C)(C(N2CCCC(N(C(c3c(C)cncc3)=O)CCO)C2)=O)CCN(C)C1=O 72329,C1(COC)(CNC(=O)CC2CCC2)CCCN1C(=O)CCN1CCC1 72330,c1(C(=O)NC2CC3(C2)CN(C(C24CC(F)C2C4)=O)C3)cccc2nonc12 72331,c1(CC)cccc(OCC(=O)NCC2CN(C(c3nccc(C)n3)=O)CC2O)c1 72332,C=CC(C)(CCOC)C(=O)NCCN(C(=O)C(c1c(C)cccc1C)O)CC 72333,c1(SCC)cc(C(=O)NC(C)CNC(C2C(C)C2C)=O)ccn1 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72611,S(=O)(=O)(c1ccccc1F)NCC1N(C(c2ccc(Cl)c(Br)c2)=O)CCC1 72612,c1(CC(=O)N(C2C3CCC2CNC3)c2cccc(Cl)c2)cc(F)cc(F)c1F 72613,C12(C(N3CC(N4CCN(C(=O)Cc5cncnc5)CC4)C3)=O)CCCC1CCC2 72614,C1(CC(N2CC(OCCC(=O)NC(C(C)C)C3CC3)C2)=O)NC(=O)NC1=O 72615,C(=O)(CCP(C)(C)=O)N(C1CCCCN(C(=O)C(c2ccc(F)cc2F)=O)C1)C 72616,c1(C(=O)NCc2c(F)ccc(F)c2Br)cc(I)ccc1[N+](=O)[O-] 72617,n1(CCC)nnnc1C1(NCc2cnoc2C)CC(n2nnnc2O)C1 72618,N1(C(C2(C)CC(=C)C2)=O)CCC2CN(C(=O)CCCOC(C)=O)C2C1 72619,Cc1cccc(C(F)C(=O)NCC2CC2CNC(C2CCCS2(=O)=O)=O)c1 72620,N1(C(=O)CCc2ncc[nH]2)CC2CC1CN2C(C1CC1c1ccc(Cl)cc1)=O 72621,N1(C(=O)C=Cc2cccc(CO)c2)CCC(CNC(C2(Br)CC2)=O)C(F)(F)CC1 72622,c1(C(=O)NCC2CCN(C(CCC3C(C)C3)=O)C2(C)C)ccc2c(c1)ncn2C 72623,Fc1cc2c(cc1Br)CN(c1nc(I)cs1)CC2 72624,c1(C(N2C(C)CC(NC(C(CC(C)C)NC(C)=O)=O)C2)=O)cc(C)nc(Cl)c1N 72625,Cn1cc(Br)cc1C(=O)NCC1(NC(=O)CNC(=O)C2CC2)CC1 72626,C(=O)(C(CNC(=O)C(O)C1CCCC1)CC(C)C)N1CC(N(CCC)CC)C1 72627,c1(N2CCC(C)(CSC)C2)nc(=N)nc(N2CCC(CCO)C2)[nH]1 72628,C(=O)(CC1=NN(C)C(=O)C1)N1CCC(C#C)(C(N2CCOC(CC(N)=O)C2)=O)C1 72629,N(C1CCc2ccc(Cl)cc21)C(C1CCCN(Cc2cn(CC=C)nc2)CC1)=O 72630,c1(-c2nc(C3CCCN(c4cn(C)nc4)C3)on2)ccc([N+](=O)[O-])s1 72631,c1(NC(=O)NC2(CC(=O)Nc3c(C)cc(F)cc3)CCC2)cc(F)c(F)c(F)c1 72632,C1(C(N(C2CCCC2)CC#C)=O)CN(C(=O)C(F)C(C)C)CC1C(C)C 72633,c1(C(N2CC(NC(CCNC(N)=O)=O)C3(C2)CC3)=O)cccc2c[nH]nc12 72634,CC1(C)CN(CCO)CCN1C(c1ccnc(Cl)c1F)C(=O)NC1CC1 72635,C1(CN(C(=O)COC2CCOC2)C)CCN(C(=O)CCN2CCC(F)C2)CC1 72636,c1(C(N2CCCC(NC(c3ccc(Br)cc3Br)=O)CC2)=O)c(Cl)cc(F)cc1Cl 72637,C(CCC(C)C(=O)N1CC(Nc2cc(C(=O)NOCCN(C)C)on2)C1)OC 72638,C1(NC(c2c(C)c(Br)n(C)n2)=O)CN(C(=O)C(C)C#N)CCC12CCC2 72639,N1(C(C(C(=O)OC)OC)=O)CC(NC(c2ccnnc2)=O)C2CCCC12 72640,N1(C(=O)CC2CC3(CC3)CO2)CCN(c2ccccc2)CC12CCC2 72641,C(=O)(C(C)(C)CCC(=O)OC)NCC(C(=O)NC(CC)C(=O)OC)C 72642,c1(N2CC(CNC(c3nc(C)nc(O)c3)=O)OCCC2)ncc2ccnc-2[nH]1 72643,c1(C(=O)NCCOCCCN(C)C(c2cc(F)n[nH]2)=O)c[nH]nc1S(N)(=O)=O 72644,N1(C(c2c(C)nn[nH]2)=O)CC2(C(=O)NC3CCC(C4CC4)C3)CC1CO2 72645,N1(C(C(C)CC(N)=O)=O)CC2CCC1CN2C(c1ncn2c1CCCC2)=O 72646,c1(C(=O)NC(C(C)C)CCN(C(=O)C(C)O)C)c[nH]c2c(Br)cccc12 72647,CCCCC(=O)NNC(=O)C1CCN(OC(=O)NC(C)(C)C)C1(C)C 72648,CC(CC(=O)N1CCCC1C1(O)CN(C(C2CCC(C)(C)CC2)=O)C1)C(F)(F)F 72649,C1(C(=O)NCC(CC=C)(C)C)CN(C(c2cnc(C)s2)=O)CC1(F)F 72650,CCN=c1[nH]c(C(=O)NCC(C2CC2)N(C(=O)Cc2nncn2C(C)C)C)cs1 72651,c1(CNC(CC=C)=O)ccnc(C(=O)NCC2C=CCCC2)c1 72652,CC1=C(C(=O)NC2CCCCN(C(C3CCCCC3C(N)=O)=O)C2)CCS1(=O)=O 72653,C1(CCN(C(CC)C(=O)NCC2COC2)C2CC2)CN(CCSC)CCS1(=O)=O 72654,CC1CCC(C(N2CC(C(N)=O)(Nc3ccccc3)C2)=O)CN1 72655,C1(NC(C(c2cccc(C)c2)C)=O)CC(F)CN(C(c2cnnc(C)c2)=O)C1 72656,CCC1=NOC(C(=O)NCCCCNC(=O)C=CCn2cncn2)C1 72657,c1(COCCO)cc(Cl)cc2cc(C(=O)O)oc12.C12CCN(C1)C2 72658,c1(C(N2CC(CC=C)(NC(=O)CCCC(C)=O)C2)=O)ccc2c(c1)CCS2(=O)=O 72659,CC(CC(F)(F)F)N(C)C(C1C2CC1N(C(=O)C(=O)N(C)C)C2)=O 72660,N1(C(CS(CC)=O)=O)CC2CC1CN(C(C1(c3ccccc3OC)CC1)=O)C2 72661,N1(C(CC(C)C2CC2)=O)CCC2(CC1)CC2NC(c1cnn2c1OCCC2)=O 72662,C1(CNC(c2c(C)cns2)=O)COCCN(C(C2(F)CCS(=O)(=O)C2)=O)C1 72663,c1(C(N(C(CNC(C(CC)N(C)C)=O)C)C)=O)cnc2c(c1)CNC2=O 72664,C1(C(=O)NC(CC(C)C)C)CCN(C(c2ccc(F)cc2)=O)C1(C)C 72665,c1(C(=O)NCC(CC)NC(c2ccccc2)c2cc(C)[nH]n2)cccc(F)c1F 72666,C=CCCCCCC(=O)NC(C)(C)CNC(=O)C(c1ccc(Cl)s1)C 72667,N1(C(CC=C=C)=O)CCC2CCN(C(c3cn(C)nc3-c3ccc(C)o3)=O)C2C1 72668,C(=O)(C(C)(C)S(C)(=O)=O)NC(CC)CCC(=O)N1CC(Cc2cccnc2)C1 72669,c1(C(=O)NCC2C(NC(CCCC(C)(F)F)=O)CCC2)sc2ccccc2c1Cl 72670,CCC(C(=O)NCCCN(C(=O)CC1(C)CC1)C)C(F)(F)F 72671,CC1OC(C)CC1C(N1CC(CC(C)NC(=O)CCC2CCOC2)C1)=O 72672,N1(c2cc(NCCCCOC)ncn2)CCN(C(c2ccco2)=O)CC1(C)C 72673,c1(C(=O)NCCN(C(=O)C(F)C2CC2)CC(C)O)c[nH]c2cccc([N+](=O)[O-])c12 72674,CC(O)C(C(=O)NC12CC1CN(C(c1n[nH]c(C3CC3)n1)=O)C2)NC(N)=O 72675,C(=O)(C1CCCc2cncn21)NC(C)(CNC(C1CCCC1)=O)C1CC1 72676,C(CN=c1[nH]c2c(c(=NC(C)CC(=O)N3CCCCCC3)[nH]1)CCCC2)OCC 72677,N1(C(C2C(OC)CCC2)=O)CC(=O)Nc2ccccc21 72678,C1(C(=O)NCC2(C)CCN(C(C=C(COC)C)=O)CC2)COc2ccccc2O1 72679,N1(C(C(C)=CC)=O)CC2(CCN(C(c3ccc(=O)n(CCF)n3)=O)CC2)C1 72680,c1(CC)cc(F)c(C(=O)NCCC2(NC(c3ccccn3)=O)CCC2)cc1F 72681,N1(C(c2n(C)cc(C#N)c2)=O)CCCC(C2CN(C(C3CC34CC(O)C4)=O)C2)C1 72682,C1(C(N2C(C(C)NC(=O)COC3(C)CCC3)CCC2)=O)CCc2c[nH]nc2C1 72683,N1(C(C=Cc2scc(C)n2)=O)CCN(C(C2CCCO2)=O)CC2(CC2)C1 72684,N1(CCC(=C)C)CC2CCCN(C(=O)COc3ccc(OC)c(C)c3)C2C1 72685,C(=O)(C(C(C)(C)C)c1nn[nH]n1)NCc1cn(CCNS(C)(=O)=O)nn1 72686,C1(CC(=O)O)(C(N(C(C(C)=O)C)CC(C)C)=O)CCSCC1 72687,c1(C(N2C3C(NC(C4(CN(C)C)CC4)=O)C(C3)C2)=O)cccc2occc12 72688,N(C(=NCC1(C)CCCO1)NC(C)C)C(C#C)CC1CCC1 72689,c1(CC)oc(C(=O)NC(C2CN(C(c3ccc[nH]3)=O)CCO2)C)cc1C 72690,S(=O)(=O)(c1ccc(CNCCC(O)CCO)cc1)N(CC=C)C 72691,N1(C(CCc2nc(C)sc2)=O)CCC(CO)(NC(C2CCOC2C(C)C)=O)C1 72692,C(CC(=O)NC(CC1CC1)C1CC1)(C(F)F)NC(c1c(C)n[nH]c1C)=O 72693,N1(C(C(C)CN(C)C)=O)CCN(C(C23CCC(CC2)C3)=O)CC1CC1CC1 72694,c1(C(=O)NCC(C)(C)CNC(=O)C(O)c2cnc[nH]2)cncc(P(C)(C)=O)c1 72695,CC1=NOC(C)(C(=O)NCCNC(=O)CCC(=O)c2ccccc2C(F)(F)F)C1 72696,c1(OCC(=O)NCc2cnc(C3C(C)C3)s2)cncc(Cl)n1 72697,C(C#CCNC(C1(CCF)CC1)=O)NC(CNC(N)=O)=O 72698,N1(C(c2n(C)nnc2CNC(=O)C(=O)NCC2CC2)=O)CCC(N=[N+]=[N-])C1 72699,C1(C2CCC2)(C(N(CCCCNC(c2ncn(C(C)C)c2)=O)C)=O)CCC1 72700,C1(c2onc(C)n2)CN(C(c2nnn(C)c2C)C(=O)NCCC2(C)CC2)CCO1 72701,N1(C(C(C2CC2)SC)=O)CC(F)(CNC(=O)C(CN(C)C)c2ccccc2)C1 72702,c1(C(=O)OC)ccc(NC(=O)C(N2CC3CCCC23)C2COC2)cc1 72703,N1(CCNC(=O)OCC2CCCC(F)(F)C2)CCc2c(Cl)cccc2C1 72704,C1(C(=O)OC)C2CCN(C(=O)C(C)CCc3cccc(F)c3)CC12 72705,C1(C(N(C2CC(NC(C(CC)COC)=O)C2)C)=O)CN2CCC1CC2 72706,c1(C(=O)NCC(CNC(C(C)SCCCC)=O)(C)F)cc(F)cnc1O 72707,CC1OCCOC1C(N1CCOCC1CC(=O)NCC1(C)CC1(F)F)=O 72708,C(C)(CCC(=O)N1CCCC1CCC(=O)NCCC12CC(CCO1)C2)OC 72709,N1(C(=O)CC2CC(Oc3ccccc3)C2)CC2ON=C(C(F)F)C2C1 72710,CCC(C)C(C(=O)NCCCCCCNC(N)=O)NC(=O)CN(C)S(N)(=O)=O 72711,CCC(CC)(CO)C(=O)N1CCC(NC(C2CCn3cncc3C2)=O)CC(O)C1 72712,Cc1nccc(C(N2CC(c3ocnc3CNC(=O)CCCF)C2)=O)c1N 72713,N1(C(C2(C)CC=CCO2)=O)CC2=C(C1)CN(C(=O)CCNC(c1cccs1)=O)C2 72714,C(CC(C(=O)NC1(C)CC(O)C1)NC(=O)CC(C)(F)F)N(C)C 72715,C1(CN(C(CCC2CCC(C)O2)=O)C)CCN(C(c2ccc(C(N)=O)s2)=O)CC1 72716,c1(C(=O)NCC(CNC(C=C(C)c2ccsc2)=O)(C)C)cc2scnc2[nH]1 72717,C1(C(=O)NC(C(=O)OCC)CC)C2CCC(C2)N1C(C1(C)CCCO1)=O 72718,C1(N(C(Cc2ncc(C)o2)=O)C)CN(C(=O)CC2CN(C)C2)CC1F 72719,CC1(C)OC2(C(N3CCOC(CNC(C4CCN(C(N)=O)CC4)=O)C3)=O)CC1C2 72720,CS(=O)c1ccc(NC(c2cc(I)cs2)c2nnnn2C2CCCCC2)cc1 72721,c1(CNC(C2(NC(C3CC3C(F)(F)F)=O)C(C)(C)C2)=O)ccccc1O 72722,CCC(CC(=O)N1CCC(NC(C23CC(CO)(C2)C3)=O)C1C)C1CCC1 72723,C1(C2CC2)(C(=O)NCC(CNC(CCC)=O)OC)CCOCC1 72724,C(=O)(CCC1=CCCCC1)N1CCN(C(CCCC#CC)=O)CC1CC(F)(F)F 72725,c1(CC(=O)NCC(C)NC(=O)CCc2ccc(Cl)nc2)cccc(F)c1 72726,C1(NC(=O)CC2CCCCC2)CC12CCN(C(c1ncc3[nH]ncc3n1)=O)CC2 72727,c1(N2CCCCC(NC(c3c(C(C)C)nns3)=O)C2)c(C#N)cccc1[N+](=O)[O-] 72728,C(c1cn(CC(CNC(=O)C(C(C)C)N2CCC(C)CC2)OC)nn1)=CC 72729,C1(CC)CCC(C)N1C(=O)CCN(C(c1cc(O)nn1C)=O)CC 72730,N1(C(C(OC)OC)=O)CCCC(CCNC(=O)CCCc2cccc(Cl)c2)C1 72731,C1(NC(C2CN(C)C2)=O)CN(C(c2cccc(CC#N)c2)=O)C2CCCCC12 72732,C(C1CCCCCC1)=CC(=O)N(CCCCN(C(C1CCC(OC)C1)=O)C)C 72733,N1(C(CNC(C)=O)=O)CCC2C1CCCN2C(c1cc(Br)cc2[nH]ncc12)=O 72734,C(=O)(CC(C)C(=O)OC)NCCC1(O)CCN(C(C2(OCC)CCOCC2)=O)C1 72735,C1(C2CN(C(=O)C(C)Cn3ccnc3)C2)(NC(Cc2c(C)n[nH]c2)=O)CC1 72736,C1(CCNC(C(F)=CCC)=O)CCN(C(=O)CNC(=O)CCC(C)C)C(C)C1 72737,c1(C(=O)NCC(CCNC(CCC(=O)OCC)=O)O)cnc(C)cc1Cl 72738,Cc1nn(C)cc1-c1cn(CCCC(=O)NCCC2CC3CCC2C3)nn1 72739,C1(OC)CC2CC1CN(C(=O)CC1CCCCC1NC(c1cncnc1)=O)C2 72740,Cc1ncnc(O)c1CCC(=O)N(C(C)CN(C)C(C1CCC2(CCC2)C1)=O)C 72741,C(CN=C(NC1CCS(=O)(=O)C1)NC1CCSC1)N1CC(C)(C)C1 72742,C(C)(C)(C(C)CC(=O)NC(C)Cc1nncn1C)NC(c1ccc(C)nc1O)=O 72743,c1(C(=O)NCCC2(C(=O)NCC3(OC)CCC3)CC2)nc(C)sc1C 72744,C(=O)(C(O)(C(F)(F)F)c1ccccc1)N1CCC(CCNC(C2(F)CC2)=O)C1 72745,C(=O)(C1CCCc2n[nH]cc21)NCCCC(C)NC(C1CC1(F)F)=O 72746,N1(C(C(C=C)O)=O)CCC(F)(F)C(CNC(c2cc(C3CC3)n(C)n2)=O)C1 72747,Cc1nnc(NC2CC(NC(c3sccc3C)=O)C2)nc1C 72748,c1(N(C2CCN(C(C(C(CC)O)C)=O)C2)C)cc(C)nc(C)c1[N+](=O)[O-] 72749,C1(C(=O)NC(COC)C)CC2CN(C(c3ncn4c3CCC4)=O)CC2C1 72750,C(C1CCCN1C(c1coc(CO)c1)=O)=CC(=O)NC(c1ccco1)C 72751,N1(C(C#CC2(CC)CC2)=O)CCCC2CN(C(C3(CO)CCC3)=O)CC12 72752,S(=O)(=O)(C1CN(C(c2cc(C3CC3)[nH]n2)=O)C1)N1CCN(C(CCOC)=O)CC1 72753,Cc1c(C(=O)NCc2ncc(C(N3CC(C)(O)C3)=O)cn2)c[nH]c1C#N 72754,CCC(C)C(O)CC(=O)N1CCOC(CC(=O)NCC(C)(F)C(C)(C)F)C1 72755,c1(C(N2CCC(CN(C(C(N3CCC(O)CC3)C)=O)C)C2)=O)cccc(Cl)c1Cl 72756,N1(C(C(C=C)(C)C)=O)CCN(C(=O)CCc2cc(OC)no2)CC2(CC2)C1 72757,N1(C(C=CC=CC)=O)CCC(NC(c2cn(C)nc2CCC(F)(F)F)=O)C1C 72758,c1(C(C)OC)nc(Cl)cc(=NC(CO)C2CC3CCC2C3)[nH]1 72759,N1(C(CSCC#C)=O)CCCC(C(C)(C)C(=O)NCc2cnn(CCC)c2)C1 72760,C1(NC(C2CC2(F)F)=O)CCN(C(=O)C=Cc2ccncn2)CC1CO 72761,C(=O)(C(F)(F)C(F)(F)F)N1CC(NC(=O)Cn2ncc(O)nc2=O)C(O)C1 72762,C1(C(N(CC(=O)N(CCCC(C)C)C2CC2)C)=O)CNC(=O)CC1C 72763,c1(NCCN=C(NCc2c(C)nn(C)c2)NC2CC2C)ccc([N+](=O)[O-])c(F)c1 72764,n1(CCC(=O)NC2C=CCN(C(CSCC#C)=O)C2)nc(O)c2ccccc12 72765,C1(C(N2C(C)(COC)CCC2)=O)CC2CCCC2N1C(=O)C1=C(C#N)CCC1 72766,N1(C(CCC=C)=O)CCC(C2CCCN2C(c2cncc(C(C)(F)F)c2)=O)CC1 72767,N1(C(Cc2nnc(C)o2)=O)CCN(Cc2cccc(C)c2O)C2CC12 72768,C(=O)(CCCC(=O)NCC1CN(C(=O)CC2CCCCN2C(C)C)CCO1)OC 72769,N1(C(c2nc(C)n(-c3ccccc3)n2)=O)CC2CC1CN(C(C1(F)CC1)=O)C2 72770,C(=O)(CS(N)(=O)=O)N(C(C)C)CCNC(=O)C(C)n1cnnn1 72771,N1(C(C(=O)NCCC(C)c2ccco2)=O)CCC(NCC(F)F)CC1 72772,C(C(CC)(CC)C(N)=O)NC(C1(CNC(CCC=C=C)=O)CC=CC1)=O 72773,N1(C(C(C(=O)O)OC)=O)CCCn2cc(Br)cc2C1 72774,c1(SC)cc(NNC(=O)NC2COc3ccc(C)cc3C2)ncn1 72775,CCCC(CNC(=O)C=C(C)C(C)C)C(=O)N(C)CCC 72776,n1(CCOCC)nc(-c2cccc(C(F)(F)F)c2)nc1C(C)OC1CCCCC1 72777,CCC(C)C(=O)C(=O)NCC1C(C)CCCN1C(c1cnn(C(C)C)c1)=O 72778,C1(NC(C(C)CO)=O)CCC2(CC1)CN(C(c1cc(C3CCOCC3)[nH]n1)=O)C2 72779,Cc1cc(C(N2CCOCC2CC(N2CCN(C(C)(C)C)CC2)=O)=O)cc(C)c1 72780,c1(C(N(CC(C)NC(C(CC)C2CCOCC2)=O)CC)=O)ncc2ccccn12 72781,C(=O)(C1=NOC2COCC12)N1CC(CC)C(NC(=O)Cc2ccc(Cl)cc2F)C1 72782,c1(OC(C)C)ccc(COC(c2ccccc2CS(C)=O)=O)c(Cl)c1 72783,C1(NC(C2(C)CC2(F)Cl)=O)CCCCN(C(C2(O)CC2)=O)C1 72784,C1(C(=O)NC(CNC(c2c(SC)csc2)=O)C2CC2)CCCCCCC1 72785,c1(NC(C2N(C(C(C)O)=O)CC2)=O)cc(Br)cnc1I 72786,C1(NC(CC=C)=O)CC2(CCN(C(c3cc4sccc4cn3)=O)CC2)C1 72787,N1(C(C(C)=C(C)C)=O)CCCC1CCNC(c1ccco1)=O 72788,N1(C(C2(C)CNC(=O)C2)=O)CC(C2CN(C(c3nccc(Cl)c3F)=O)C2)C1 72789,N1(C(c2cc(C)cc(F)c2)=O)CCC2(CC2)CC1C(=O)NC(C)C(C)(C)O 72790,c1(C(=O)NCC(C)NC(Cc2c(C)cco2)=O)cc2c(n1C)CCOC2 72791,C(=O)(CC(CC(C)C)NC(=O)CCn1cnc(=N)[nH]1)Nc1cn(CC)nc1 72792,N1(C(c2ccc(OC)cc2O)=O)CC(C2CC2)C(F)(C(=O)O)C1 72793,C1(C(N2CC3C(NC(c4c(SC)cccc4)=O)(C3)C2)=O)CCN(C)S1(=O)=O 72794,C1(NC(CNC(CC)C)=O)CCCN(C(=O)C=CCN2CCCC2)CC1 72795,c1(C(N2CC(NC(c3ncc(C)c(C)c3)=O)C(C)C2)=O)ccc2c(c1)NCCC2 72796,C=C(C)C(C)(C)C(=O)NC1CCCC(CNC(c2ccc(C(F)(F)F)nn2)=O)C1 72797,C1(C(=O)OCC)CN(C(=O)C=CC(=O)NCC2(F)CCCC2)CC12CCOCC2 72798,C1(N(c2cccc(C(C)C#N)c2)C(c2c(C)noc2)=O)CCNCC12CC2 72799,c1(C(c2n(CC=C)nnn2)NCC(C2CCCCC2)OCC)nccc(Cl)c1C 72800,Cc1cnc(C(=O)N(CC(C)(C)NC(C2(n3cccc3)CCCC2)=O)C)c(C)c1 72801,C1(CC(=O)N(CCCCN(C(=O)Cc2cnco2)C)C)OCCC1(C)C 72802,S(=O)(=O)(c1cccc(C(=O)NC(c2ncccn2)(C)C)c1)N(C(CC)C(N)=O)C 72803,c1(C(=O)NC2CC3(CN(C(CC=CC)=O)C3)C2)cc([N+](=O)[O-])ccn1 72804,N1(C(CCCC#C)=O)CCOCC(NC(=O)CC(C)Cc2ccc(F)cc2)C1 72805,C1(C(=O)NCC2(O)CN(C(CNC(C(CC)C)=O)=O)C2)CNC(=O)C(C)(C)C1 72806,CC(C)C(F)(CNC(C1CCCC12CCC2)=O)C(=O)N(C)CC1CCOC1C 72807,C(=O)(C(C)(C)CC(=O)NC1COCCC1C(N1CCCC(F)(CO)C1)=O)OC 72808,c1(C(=O)NC2C(OC)CN(C(c3cccn3C)=O)C2)ccc2c(N)nccc2c1 72809,N(C1COc2cc(Br)cc(C)c21)C(=O)NCc1ccc(-n2ccc(C)n2)c(F)c1 72810,C=CCCC(C(=O)NC1CCCN(C(C)C)C1)NC(=O)CC1CCCSC1 72811,N1(N(C(c2nc(C(C)C)on2)=O)C)CCCC(n2cc(C(C)(C)F)nn2)CC1 72812,c1(C(COC)(C2CCCC2)NCC2CC2C)nnnn1Cc1ccccc1 72813,CC1C(C)N(C(=O)CC23CCC(CC2)OC3)CCN1C(=O)C(C)OCCN(C)C 72814,C1(N)(C(=O)OC2CCCN(C(C)C)C2)CCCC(C)CC1 72815,c1(C(=O)NC2CC2)cnn2cccc(-c3ccc(OCCCO)cc3)c12 72816,c1(C(=O)NCCC2CC(NC(CC#N)=O)C2)ccc2c(c1)S(=O)(=O)NC2 72817,C(=O)(C(C)(C)CCC#N)NC1C(OCC)COC1 72818,c1(N(C(c2cc(CC3CCCCC3)on2)=O)CCO)ccc2c(c1)OCO2 72819,C(=O)(C(O)CC[S+](C)C)N(CCCNC(C(C)OCCC=C)=O)C 72820,C1(OC)CC2(C1)CN(C(=O)CC(O)CNC(=O)C(c1cnn(C)c1)O)C2 72821,C(=O)(NN1CCCC1C(=O)N(C1CCCC1)C)C1CC(N(C)C)C1 72822,c1(OC)cc(C2(C(=O)NCC(C)(O)CNC(=O)CC3CC(F)C3)CC2)ccc1C 72823,c1(COCCOC2CCN(C(C(c3ccccc3)SC)=O)C2)ccnc(F)c1N 72824,N1(c2cc(C)ncn2)CCCCC(NC(=O)Cc2c(F)cccc2F)CC1 72825,c1(CCC(=O)NC2CCC(CNC(C3(C)CC3)=O)C2)cc(Cl)ccc1Cl 72826,n1(C(C(=O)NC(C(C)C)c2nn[nH]n2)C)cc(C(C)CC2CCC2)nn1 72827,CCC(C)(O)CCNC(C1(NC(C2C3CCCOC23)=O)CCSC1)=O 72828,Cc1ccc2ncc(C(N3CCCC(NC(c4coc(C)n4)=O)C3)=O)n2c1 72829,c1(CC(N2CC(O)(CCNC(C(C)O)=O)C2)=O)cccc2c1oc1ccccc21 72830,C(=O)(CCCCCF)NC1C(C)CN(C(c2cnc(C(C)(C)C)[nH]2)=O)C1 72831,C1(C(N2CC(C)C(CC(=O)Nc3cncc(Cl)c3)C2)=O)CCCCCN1C 72832,CC12CN(C(=O)Cc3ncc(Cl)s3)CC1CN(C(c1coc(C(F)F)n1)=O)C2 72833,c1(C(=O)NC(C)CNC(=O)Cc2n[nH]c(O)n2)cccc(-c2ccoc2)c1 72834,C1(NC(c2c(OC)ccs2)=O)CCCC(C(=O)NCc2cnco2)C1 72835,C(CNC(=O)CC1CC1)(C(C)C(C)C)NC(C(=Cc1ccncc1)C)=O 72836,c1(CC)cc(C(N2CC(CNC(=O)C(C)C)(OC)C2)=O)n[nH]1 72837,c1(N2CCCC(NC(C(c3cn(C)nc3)O)=O)CC2)ncnc2c1ncn2C1CC1 72838,N1(C(C(C)=CC2CC2)=O)CCC2(NC(c3conc3C)=O)CC2C1 72839,C1(C(=O)OC(C)(C)C)CCN(C2CN(C(C)Cn3cncn3)C2)CC1 72840,c1(C(=O)NCC2(F)CC(CNC(C(CC(=C)C)C)=O)C2)cncc(S(C)(=O)=O)c1 72841,c1(C(=O)Nc2c(NCC3CCC(C)(C)CO3)cccc2)c(Cl)cccc1[N+](=O)[O-] 72842,c1(SC2(C(=O)NC(C)CN(C)C(C3CCC3C(F)(F)F)=O)CCC2)ccccc1 72843,N1(C(CCNC(C#CC(C)(C)O)=O)=O)CCC(C2CC2)C(O)C1 72844,CC(C)CCCCCC(=O)NCC1C2CC1N(C(c1coc(Cl)n1)=O)C2 72845,Cc1ccc(CC2COCCN(C3CCNCC3)C2)c(C)c1.c12noc(n1)C2 72846,c1(CC(=O)NC2CC(CNC(C=CC(C)C)=O)OCC2)ccc(C(F)F)cc1F 72847,c1(CN2CCC(NC(CC(CC)O)=O)(CO)CC2)c(Cl)nc(SC)nc1Cl 72848,c1(CN(C(=O)CSc2nc[nH]n2)CCNC(CC2(SC)CC2)=O)ccccc1 72849,CC1CN(C(=O)CC(C)CN(C)C)CCCN1C(=O)CCn1cccc1 72850,c1(C(=O)O)cccc(Cl)c1C1CCN(C(c2ccn(C(F)(F)F)n2)=O)CC1 72851,N1(C(C2(SC)CCC2)=O)CCCC(C(C)C(=O)NCCN(C)C2CC2)C1 72852,C(CN=c1[nH]c(N2CCN(CC(F)(F)F)CC2)nc2c1CCC2)SC 72853,c1(C(c2nnnn2CCC2CC2)NC(C(=O)N(CC)CC)C)ncc(C)s1 72854,c1(N2Cc3c(ccc(OC)c3)CC2)nc2c(c(=NCCCP(C)(C)=O)[nH]1)COC2 72855,c1(OCC)cccc(C(N2CC(O)CC2C(=O)Nc2nc(C#N)cs2)=O)c1 72856,C1(NC(C(C)(C)F)=O)CCN(C(=O)CSCc2cccc(Cl)c2)CCC1CO 72857,c1(CNC(c2ccc(-c3cccc(Br)c3)cc2)C)cccnc1F 72858,Cc1cccc(OCC(N2CC(NC(=O)CSCc3cccnc3)C3CC23)=O)c1 72859,c1(C(C)C)ncc(NC(=O)C(C)C(C)NC(=O)Cc2ccoc2)cn1 72860,c1(OCC)ccc(Br)cc1CN(C=O)Cc1ccc(Br)c(C)c1 72861,c1(CN2CC(F)(C(=O)NC(c3ccc(O)cc3)C)C2)cccc(I)c1F 72862,C(CC)(CCCC(=O)N(C)CP(C)(C)=O)NC(C1C(=C)C1C(=O)OC)=O 72863,CCCCCC(C)CC(=O)N1CCC(NC(=O)CCc2ccc(O)nn2)C(F)C1 72864,C(=O)(CC(C)CC(C)(C)C)N1C(C(N(C(C)C)C)=O)CSC1 72865,C(=O)(CC(F)(F)Cl)NCC(c1ccc(F)cc1)NC(CCNC(CC(C)C)=O)=O 72866,CC1Cc2cc(C(=O)NC3COCC3NC(=O)Cn3cnnc3)ccc2O1 72867,C#Cc1nccnc1NC(C1CCCN1C(=O)CCNC(c1ccc[nH]1)=O)=O 72868,N1(C(c2n(CC)ncc2)=O)CC(NC(c2cc(C)cc(C)n2)=O)CC(O)C1 72869,N1(C(COCCCC#C)=O)CC2CCC(CNC(=O)C(O)CC(C)C)(C2)C1 72870,CC(Cl)(Cl)C(=O)N1CC(C(N)=O)(CNC(c2ccc(C(N)=O)o2)=O)C1 72871,C1(CNC(CC2N(C(C3CC(N(C)C)C3)=O)CCCC2)=O)OC(=O)NC1(C)C 72872,c1(NC(c2n(C)cc(NCc3ccc(Br)[nH]3)n2)=O)ccc(Br)cc1C(C)(C)C 72873,c1(OC)ccc(C(=O)NC2CCN(C(c3cc(C)ccn3)=O)C(C)C2)c(F)c1Cl 72874,C1(C(N2CCN(C(C3CCC3)=O)CC2)=O)C2CC(O)C(C2)N1C(=O)C1CC1 72875,N1(S(CC)(=O)=O)CCC(C(=O)NCc2ncc(-c3cccc(Cl)c3)o2)CC1 72876,N1(C(C2(c3c(C)cccc3)CCC2)=O)C2CCCC1CC(NC(=O)C(C)(C)F)C2 72877,c1(C(N2CC(C(=O)NC3CC3)C2)=O)cnc(CNC(=O)CC2CCC(=O)C2)nc1 72878,N1(C(C2CCC(CC)C2)=O)CCN(C2CCN(C(=O)CN(C)C(C)C)CC2)CC1 72879,c1(C(=O)N(CCCn2cc(-c3cncc(Cl)c3)nn2)C2CC2)c[nH]nc1[N+](=O)[O-] 72880,C1(CNC(C(CC)F)=O)CC2(CCN(C(C34CCC(F)(CC3)C4)=O)C2)CO1 72881,c1(OC)ccc(C(O)C(N2CC(O)(C(C)NC(=O)Cc3cnoc3)C2)=O)cc1 72882,C1(C(=O)NCCCCN(C(COCCN(C)C)=O)C)CCCCN1C1CCCC1 72883,c1(C(=O)NC2CCCC(CC(=O)NCCOCC)C2)c(C)cnnc1O 72884,c1(C(N2CC(NC(c3n(CC)ncc3)=O)CC2(C)CC)=O)ccc2n[nH]cc2c1F 72885,C(=O)(CCCC(C)(C)C)NC1C(CN(C(c2ccc(CNC(C)=O)o2)=O)CC)C1 72886,C(C(CC1CCCC1)C(=O)Nc1ccc(C2CC2)cc1)NC(C(COC)C)=O 72887,C1(CCCNC(C2C(C)C2)=O)CCCN1C(C1CCC(=O)N1)=O 72888,C12(CNC(C3CC4(CC4)C3)=O)CCCC1CCN2C(c1cc2c(s1)CCC2)=O 72889,C(=O)(CC(C)(C)C1CC1)NCCCC(C)NC(=O)CC1C=NN(C)C1=O 72890,CC1CCCn2cc(C(N3CCCC4(NC(C5CCCCC5)=O)CC4C3)=O)nc21 72891,c1(C(N2CC3C(CNC(c4c(CC)onc4C)=O)(C3)C2)=O)ccc(F)cc1O 72892,C1(COCC)CCN(C(=NCSC)NCC2CCCOC2c2ccccc2)C1 72893,N1(CCCNC(c2cccn(C)c2=O)=O)CCC2(CCCCC2)CC1 72894,C1(NC(C(C)=CC2CC2)=O)CC(C(=O)N(C)Cc2cnccn2)C1(C)C 72895,C#CCCCC(C)C(=O)N1CCC2(CC2NC(=O)C(c2ccccc2F)C)C1 72896,C=C(C)C(C)(C)C(=O)N1CC(CO)(NC(=O)CN2CCCC2CO)C1 72897,CCC(C)CCCC(=O)NCCC1CC(C(=O)NCCOCC(N)=O)C1 72898,CS(=O)(=O)c1ccc(C=CC(=O)NC2CCN(C(=O)CC(F)F)CCC2CO)o1 72899,Cc1ccc(C(=O)NC2CCC2NC(c2cc(O)ncc2Br)=O)c(F)c1 72900,N1(C(CC2CCN(OC)CC2)=O)C2CCC1C(F)C(NC(=O)C(C)(C)CO)C2 72901,C1(C(=O)N(c2c(C)nco2)CCO)C2CN(C(c3coc(C(N)=O)c3)=O)CC12 72902,N1(C(=O)C2=CCCCC2)CCC2CCCC12C(=O)NCC12CCC(CC1O)C2 72903,C1(CNC(=O)CN2CCCS2(=O)=O)C(C2CC2)CCN1C(=O)Cc1ccc(Cl)s1 72904,C(=O)(CC(CC1CC1)NC(=O)CC(O)CN(C)C)NCCc1scc(C)n1 72905,N1(C(CCCC#CC)=O)CC(C2CCN(C(c3ccoc3)=O)C2)C1 72906,N(C1CN(C)Cc2ccccc21)C(=O)Nc1c(OC)ccc(C(=O)OC)c1 72907,CC1(C)CCCC1CCCNC(=O)NC1(Cc2ccc(Cl)cc2)CC1 72908,N1(C(C(C(C)C)O)=O)CC(NC(C23CC(c4ccccc4)(C2)C3)=O)CCC1C 72909,c1(C(N2C(C(=O)NCC3C(C(=O)OC)C3)CNC(=O)C2)=O)cccc2cncn12 72910,c1(C(N2CCC(CNC(CC(C(F)(F)F)OC)=O)C2)=O)cc(O)c2sccc2c1 72911,O=C1CCC(N=c2[nH]c(NC3C4CCCC34)nc3c2CCCC3)CN1 72912,C1(NC(CC(=O)OCC)c2ccccc2)CCCN(CCCNC(C)=O)CCO1 72913,C1(CCC(=O)NC(=O)OC(C)(C)C)CCC(NC2CC(C(=O)O)(CF)C2)O1 72914,C1(NC(c2ncc(OCC)nc2)=O)CC2(CCN(C(C3(CC)CCOC3)=O)C2)C1 72915,c1(C(N(CC(CC)NC(=O)CNC(C)=O)C)=O)cc(Br)cc(C)c1F 72916,C1(CNC(C2N(C(CSC)=O)CC=CC2)=O)CCCC2(CC2)C1 72917,C12(NC(CCCCCNC(C)=O)=O)CCC(CN(C(C3(F)CCOC3)=O)C1)C2 72918,C1(CC)CC(C(N(C)CP(C)(C)=O)=O)CCN1C(=O)COc1cnn(C)c1 72919,C1(C(=O)Nc2cccc(OC)n2)CCN(C(c2cncc(F)c2)=O)CC1O 72920,N1(C(c2cc(OCCC)c(F)cc2)=O)CC(C(=O)NC)CC(F)(F)C1 72921,CCC(O)CCNC(=O)CC1(CNC(=O)Cc2ccsc2C)CC1 72922,C1(NC(C2C(C)C2)=O)CC12CCN(C(c1ccc(C(F)F)cn1)=O)C2 72923,N1(C(C2C(=C)CC2)=O)CCCC2(NC(c3coc(COC)n3)=O)CC2C1 72924,c1(C(N2CC(C(C)NC(CC3(C=C)CC3)=O)OCC2)=O)c(CC)nn(C)c1Cl 72925,c1(SCC(=O)NC23CC(NC(C4CCC(CC)C4)=O)(C2)C3)nnc2ccccn12 72926,c1(C(=O)NC(CC)CN(C)C(c2cc(Cl)n(C)n2)=O)cccc(F)c1C#N 72927,C(C(CC)CC)(c1n(CCOC)nnn1)NC(c1cccc(OC)c1)C 72928,C1(C(=O)NC2C(C(N(C(C)C(F)F)C)=O)CCC2)CCCC(=O)N1C 72929,C(=O)(C1=CCCOC1)NC(C(C)(C)C)CNC(=O)COCC1CCCOC1 72930,C(N1CCOC(C2CC2)C1)N1CCC(C)C1=O 72931,c1(C(=O)NC(CO)C2CC2)cn2c(n1)CN(C(c1c(F)ccc(O)c1F)=O)CC2 72932,c1(C(=O)NCCC2CCCN(C(c3cnc(O)s3)=O)C2)ccc2cccnc2n1 72933,N1(CC(=O)N(C(C)CNC(C2CC23CCOC3)=O)C)CCS(=O)(=O)CC1 72934,N1(C(c2cnc(C)[nH]2)=O)CCN(C(C2CC=CCO2)=O)CC1CS(C)(=O)=O 72935,CCC(CC)C(C)C(=O)NC(C)(CNC(=O)Cc1ccc(F)cc1C)C1CCC1 72936,CN1CCC(C(=O)NC2CC2NC(=O)C=Cc2cccc(CO)c2)S1(=O)=O 72937,c1(C(N2CC(C(C(=O)N(C)CC3CCC(=O)N3)O)C2)=O)ncncc1Cl 72938,N(C1CC2(CN(C(C3CC(C)N(C)C3)=O)C2)n2ccnc21)C(C(C(=C)C)(C)C)=O 72939,O=C1CCC(NC(=O)CC2CC3(CC3)CN2C(c2ccc(F)cn2)=O)C(=O)N1 72940,N#CC1CCCC1NC(C1CCCN1C(=O)CCC1CCC(=O)C1)=O 72941,C(CCCCC(=O)NCCCCSC(F)(F)F)n1cc(-c2c(C)nccc2)nn1 72942,C1(NC(C(=C)F)=O)CCN(C(c2cc(Br)ccc2OC(F)(F)F)=O)CC1F 72943,Cc1nc(SC(F)F)sc1CC(=O)NCCC(C)NC(=O)CCC(C)N(C)C 72944,CN1C(=O)CN(CC(N2CCN(C3CN(C(=O)C4=C(Cl)CCC4)C3)CC2)=O)C1=O 72945,c1(C(=O)NCC(CNC(CNS(NC)(=O)=O)=O)F)ccc(C(F)(F)F)nc1 72946,S(=O)(=O)(c1ccc(C#N)c(N(CC(C)OC)C)c1)N1CC(CC)C2(C1)OCCO2 72947,c1(C(=O)NC(c2ccnn2C)C)cnc(N)c([N+](=O)[O-])c1 72948,Cc1c(C(N2CCC(CNC(=O)CC(=O)NC3CC3)CC2)=O)sc(Cl)c1Cl 72949,C(=O)(CCS(=O)(=O)C(F)(F)F)NCC1N(C(c2cc(C(C)=O)sc2)=O)CC=C1 72950,N1(C(C2(CN(C)C)CCCC2)=O)CCCC(CO)(NC(C2CC(CF)C2)=O)C1 72951,C(CC(F)F)(C(=O)N(C)Cc1ccsc1)NC(C1C(C)C1)=O 72952,C1(C(N2CC(C)(CC)C2)=O)C(C2CC2)CCN1C(C1COCCC1C)=O 72953,C1(NC(CNC(=O)NC)=O)CCC2(CC1)CN(C(=O)C(C)(CC)CO)CCO2 72954,N1(C(C(C(=O)OC)C)=O)CCC(C(=O)N(C)CCF)=C(F)C1 72955,O=C1NCC2(CCN(C(c3cccc4ccoc34)C(=O)NCc3ccco3)C2)O1 72956,C(=O)(C#CC(=O)N(C)C)NCC(C)(C)NC(CCc1c(C)ncs1)=O 72957,c1(C(=O)NCCCC(C(=O)OC)O)nc2ccccc2nc1O 72958,c1(CC(=O)NC2C(CNC(C(CCC)C)=O)CCCC2)sc2ccccc2c1C 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72976,c1(CC(=O)NC2CCC2NC(C2CC(=C3CC3)C2)=O)ccsc1[N+](=O)[O-] 72977,C1(CC)(NC(=O)CCCc2ccncc2)CCN(C(=O)C(O)C2CCCC2)CC1 72978,c1(C(=O)NCCCn2ccnc2)cc(O)ncc1Br.c12cccc(c1)C2 72979,C1(NC(C(CC)NC(N)=O)=O)CCN(C(c2ccc(N)c(F)n2)=O)C12CCC2 72980,C1(NC(c2ccc(Br)cc2)=O)CCC(O)CN(C(c2sccc2F)=O)C1 72981,c1(CC)ccc(OC)cc1.C1(NC(N(CC(O)(COC)CO)C)=O)CC=CCC1 72982,c1(CNC(C2Cc3nccnc3C2)=O)cc2n(n1)CCNC2 72983,c1(CC(=O)NC2C(NC(c3cncc(C)n3)=O)C2)ccc(C)c(F)c1 72984,Cc1cc(Br)ccc1NC(=O)C(C1CCO1)N(c1ccsc1)C 72985,c1(C(=O)NCC2C(C)CCCN2C(C2CC(O)C2)=O)cnn2c1CCCC2 72986,c1(C(N2CCC(OC)(CNC(=O)C(CO)N(C)C)C2)=O)c[nH]c2cc(F)ccc12 72987,C12(NC(c3c(N)c(Cl)ccc3)=O)CCCC1CN(C(=O)CC1(O)CCOCC1)C2 72988,CC1CC(C#N)(C(=O)NCC2(CNC(=O)CC3CCC(=O)NC3)CC2(F)F)C1 72989,c1(CNC2C(C(=O)NCc3cccc(C)n3)C2)cc(F)c(Cl)nc1Cl 72990,O=[N+]([O-])c1cc(-n2cc(C3(OC(F)(F)F)CCNCC3)nn2)c(Br)cc1F 72991,C(=O)(NNC(=O)CCCn1cc(C2CCCO2)nn1)c1c(O)ccc(OC)c1 72992,CS(=O)CCC(O)C(=O)NCC12CC(NC(=O)CCC3CC3)(C1)C2 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73010,c1(OC)cc(CCNC(=O)N(C(C)CC(C)C)C)ccc1O.C1C(=O)N1 73011,N1(C(CCC2(C)N(C(Cc3cn(CC)nc3)=O)CCC2)=O)CCC(C)(C2CC2)C1 73012,N1(C(CN(C)CC)=O)CCCC(CNC(=O)CCOc2ccccc2C)C1 73013,C(CN=C(NCC(C)(COC)COC)NC1CCNC(=O)C1)OC 73014,N12CC(C(C)C1)NC(=O)CSCC2=O.C1(C(=O)N)CCCN1c1ccncn1.CO 73015,c1(NC(=O)Cc2nc[nH]n2)ccc(Cc2cn(CCCCCO)nn2)cc1 73016,c1(C(=O)NC(C(C)C)C(N2CCC(N=[N+]=[N-])C2)=O)coc2c1COC2 73017,C1(CC(=O)NCC(C2CCCCC2)NC(CC(=O)OC)=O)CCC(OC)CC1 73018,CCCCC(CC)CC(=O)N(CCC(=O)NCc1c[nH]nc1C)C1CC1 73019,C=CCCCCCCC(=O)NC1CCN(C(c2coc(O)n2)=O)C(C2CC2)C1 73020,c1(C(N2CC(C)C(NC(=O)CC3CCC(C)(C)CC3)C2)=O)onc2ccccc12 73021,C1(NC(C2CCC(C)(C)O2)=O)CC2CCC(C1)N2C(=O)C(C)(C)c1cncs1 73022,CC1CCc2[nH]c(=NC(C)c3cnn(C)c3)[nH]c(=NCCCCC(F)(F)F)c2C1 73023,C(C)(C(=O)NOC(CC(C)C)C(=O)NC)(N(C(C(CC)C)=O)C)C1CC1 73024,C1(CNC(C2CC(C)(C)C2)=O)CC(O)CN1C(c1ccnc(C2CC2)c1)=O 73025,C1(OCC#C)CCN(C(=O)CCC2CC2C(=O)OC)C1 73026,C(=O)(CS(=O)(=O)N1CCOCC1)NCC(C)N(C)C(c1ccc(C(C)O)cc1)=O 73027,c1(NC(=O)NC2CCN(C)CC2)cnc2ccnn2c1O 73028,N#Cc1cncnc1N1CCC(NC(c2ccc(C3CC3)cc2)=O)C(F)C1 73029,c1(OC)c(CNC(=O)C(=O)NC2CN3CCC2C3)c(C)nn1C 73030,C=CCC(C)(C)C(=O)NCC1(NC(c2cccc(-n3ccc(CC)n3)c2)=O)CC1 73031,C1(NC(C=NOC)=O)CC2CCC(C1C)N2c1cccc(F)c1C#N 73032,c1(C(=O)NC2CCCN(C(c3cncc(SC)c3)=O)CC2)cc(C)c(C)nc1C 73033,c1(CC(N2CCN(c3cc(C)ncn3)C(CC#N)C2)=O)ccc2c(c1)OCO2 73034,C(=O)(C1=CCC2CCC1N2C(C1CCSC1)=O)NC(C#C)(C)C1CCC1 73035,N1(C(C)=O)CCN(C(=O)C(c2ccc(C)cc2)c2cnn(C)c2)CC1C 73036,c1(NCC(C(C)(C)C)OC)[nH]c(=NCc2cc(F)c(Br)cc2F)nc2scnc12 73037,N1(C(C(CC(=C)Cl)NC(=O)CNC(=O)C(C)(C)C)=O)CC(C)(C)C2COCC12 73038,C#CCC(CC(=O)N(CC(C)NC(C1CCC(C)(O)CC1)=O)C)c1ccccc1 73039,C1(C(=O)NCC2C(C)(C)COC2)CN(C(C2CCCC2)=O)CC1(F)F 73040,c1(NC(C2(C)CN(C(CC=C=C)=O)C2)=O)cc(O)ccc1OC 73041,CC1CC(NC(C2CC3CCC2O3)=O)CN(C(=O)Cn2cnc([N+](=O)[O-])c2)C1 73042,N1(C(C(C=C=C)C)=O)CC(CC(=O)NC(c2nc[nH]n2)CO)CC1(C)C 73043,C1(C)(CNC(C2C(=C)CC2)=O)CCCN1C(C1(c2cccc(N(C)C)c2)CC1)=O 73044,Cc1cc(Cl)c(C(=O)NC(CNC(=O)CC(C)c2ccccc2)CO)s1 73045,N1(C(C2C(OC)C2)=O)CCC2CN(C(c3cnc(OC)c(C(F)(F)F)c3)=O)CC12 73046,C1(F)(CNC(C(C)(C)c2cscn2)=O)CCC(NC(=O)C(N)=O)C1 73047,c1(NC(=O)C(=O)OC)ccc(CN(C(C)C(C)C)CC)c(O)c1 73048,C(=O)(C(O)CC(C)C)NC(COC)CC(=O)N1CCOC(C(N)=O)C1 73049,c1(C(N(C2CN(C(CN3CCC(OCC)C3)=O)C2)C)=O)cc2c([nH]1)CCCC2 73050,c1(C(=O)NC(CN(C(=O)CC2CCNC2=O)C)CO)ccc(SC2CC2)cc1 73051,C1(NC(=O)CC2(O)CCOC2)CCC2CC1CN2C(c1nc(F)ccc1Cl)=O 73052,c1(CC)oc(C(=O)NC(C)(CNC(c2cccc(C)c2)=O)C2CC2)cc1C 73053,c1(CC(N2CCC(C)(CCNC(c3ccc(C)cc3)=O)C2)=O)cccc(C#N)c1 73054,c1(-c2cn(CC(=O)NCC(CN(C(CCC)=O)C)O)nn2)cccc(SC)c1 73055,c1(C(=O)NC2C3CN(C(c4[nH]c(=N)sc4)=O)C(C3)C2)cc2cc(F)c(F)cc2[nH]1 73056,N1(C(C(C(C)C)OC)=O)CC(CO)C2(CCN(C(=O)CC(C)CC(C)C)CC2)C1 73057,N1(C(C)=O)CCCCC1CC(=O)NCC1(F)CC(NC(c2[nH]nnc2C)=O)C1 73058,N1(C(c2n(CC)ncc2)=O)CCCC(CO)(NC(=O)CN(c2ccncc2)C)C1 73059,C1(C(N(C)CC2CCCC(C)C2)=O)CCCN(CCC(C)N(C)C)CC1 73060,N1(C(c2n(C=C)ncc2)=O)CC(NC(=O)Cc2ccc(OC)cn2)CC12CCC2 73061,CC(O)C(C)C(=O)N1CC(CO)C(CO)C1 73062,C(=O)(C(C)(C)CC#N)NCCCCC(C)NC(=O)COc1ccc(F)cn1 73063,c1(C(=O)NCC(C)CNC(=O)C(C)NC(N)=O)ncccc1[N+](=O)[O-] 73064,Cc1nccc(Cl)c1C(=O)NC1CC(F)CN(C(c2ccnn2C(C)C)=O)C1 73065,N1(C(C(CCC)CNC(=O)C(C)OCCOC)=O)C(C)CC2CCCC12 73066,CC1CC(CC(=O)N(C)CC2CN(C(C3CCCCC3C)=O)CCO2)C(C)O1 73067,c1(C(N2C(COC)CN(C(C3(Cl)CC3)=O)CC2)=O)cccc2c1NCC(C)C2 73068,N1(C(C(C)C)=O)CC2(C1)CN(C(c1cccnc1-c1ccccc1)=O)C2 73069,CCCCC(C)(F)C(=O)NC1CC1C1CCOCC1 73070,c1(C(C(=O)OC)NC2CC(=O)NC2=O)cc(Cl)cc(Br)c1 73071,Cc1c(C(N2CCC(C(C)(O)CNC(C3CC3C(N)=O)=O)CC2)=O)nn(C)c1N 73072,C1(NC(=O)CCc2cccs2)CCCC1CC(=O)NCCc1ccsc1 73073,C(=O)(C(CNC(C)=O)NC(C1CC1(Br)Br)=O)OC 73074,C1(C(N(C2CCN(C(c3nncs3)=O)C2)CCO)=O)CC2C=CC1CC2 73075,N1(C(CCNC(=O)Cn2ccccc2=O)=O)CC2C3C=CC(O3)C2C1 73076,C(=O)(CC1=CCOCC1)NC1CC(CNC(CC2(COC)CC2)=O)CC1O 73077,Cc1cnc(N2CC(NC(=O)CC(=O)NCC(F)(F)F)CCC2C)nc1O 73078,c1(OC)c(OC)cc(C(=O)NCC(C)(C)NC(C2CC3(C2)CC3F)=O)cc1Cl 73079,N1(C(C(C=C)OC)=O)CCC(CNC(c2cnncc2NC)=O)C1(C)C 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73098,C1(NC(C=C(Cc2c(OC)cccc2)C)=O)CC2CC(NC(=O)C=C(C)C)CC12 73099,N1(C(C(CCN(C)C)O)=O)CC2C=CC1C(C(N1CC(NC(N)=O)C1)=O)C2 73100,c1(CN2C(C(N3CCC3CO)=O)CC3CC32)cc(F)c(O)c(F)c1 73101,N1(C(C2(C)CS(=O)(=O)C2)=O)CC2=C(C1)CN(C(c1cnn3c1SCC3)=O)C2 73102,N1(C(C2CSC2)=O)CC2OCCN(C(c3cc(Cc4cccs4)on3)=O)C2C1 73103,N1(C2CC3(NC(c4ccc(OC(F)F)nc4)=O)C(C2)C3C)CCSCC1CCO 73104,N1(C(CNC=O)=O)CC(n2cccc2)C1 73105,c1(CC)ncc(C(=O)N(C)CCN(C(=O)CC2CC2(C)C)C(C)C)o1 73106,c1(C(=O)NCC(C(C)C)(C)C(C)C)cccc(N=c2cncc[nH]2)c1 73107,CC(C)(F)CCC(=O)NCC1CCCC1NC(c1cnoc1-c1ccccc1)=O 73108,CCCCCCCCCC(=O)NC(C)C(C)NC(C1CC=C(C)CC1)=O 73109,CCC(CS(=O)(=O)c1ccc(C)c(C)c1)NC(=O)CS(=O)(=O)c1ccccc1F 73110,c1(OC(=O)NCC(C(C)C)NC(C=CC)=O)cnc(O)n(-c2ccccc2)c1=O 73111,N1(C(Cc2c(C)noc2C)=O)CC2CCCC2(NC(c2cc(C(F)F)no2)=O)C1 73112,N1(C(C(C)=C2CCOC2)=O)CC2CCC(CNC(=O)C(C3CCCCC3)C)C2C1 73113,N1(C(c2cc(C)no2)=O)CCC(CC(=O)NCc2cnn(C(C)C)c2)C1(C)C 73114,C1(C(N2CCC(CNC(COC(CC)(C)C)=O)C2)=O)CCN(C2CC2)S1(=O)=O 73115,Cc1cc(Cl)cc(Br)c1NC(C1CN(C(C2CC(C)(C)C2)=O)CC(F)(F)C1)=O 73116,CCCCC(CNC(=O)Cc1csc(S)n1)NC(c1cc(O)no1)=O 73117,C=CCC(CC(F)F)C(=O)N1CC2CC(C1)N(C(=O)CC1CCCN1C)C2 73118,N1(C(c2c(C)coc2)=O)CCCC(C2CN(C(=O)CCCc3ccncc3)C2)C1 73119,C1(C(C)=O)CN(C(c2cc(C)cc(O)c2)=O)CCN1C(=O)CNC(N)=O 73120,S(=O)(=O)(c1ccc(NCCSC(F)(F)F)cc1Cl)NC(C)(C)CCO 73121,C1(CNC(CCCCN(C)C)=O)CC2CCC1N(C(c1nc(Cl)sc1Cl)=O)C2 73122,CC1CN(C(c2cc3n(n2)CCCC3)=O)CCN(C(=O)COC(C)(C)C)C1 73123,CCC(CNC(=O)C=Cc1ccsc1)(CC)NC(=O)CNC(=O)CCC 73124,c1(OC)cccc2ncnc(N3CCCCC3CCNC(C3(OC)CCC3)=O)c12 73125,CC1CC(CCC(=O)N(C(C(=O)NCCSC(F)F)C2CC2)C)C1 73126,C1(CNC(CN2CCC(C(=O)NC)C2C)=O)CCCCCN1Cc1ccccc1 73127,c1(C(N(CC(CC)NC(c2ccc(CO)s2)=O)C)=O)c[nH]nc1Br 73128,c1(C(=O)NCC2(CN(C)C(C3CCC4CC34)=O)CC2)cc(S(=O)(=O)N(C)C)c[nH]1 73129,C1(C(c2n(CC=C)nnn2)NCc2cncn2CCC)CCC2(CC1)CC2 73130,C(C(CC)N=c1[nH]c2ncc(Cl)cc2o1)NC(COCCCC)=O 73131,C=CCCCC(=O)NC1CCCCC1CC(=O)NCC1(OCC)CN(C)C1 73132,C1(C(=O)NC(C)C(F)(F)F)(C(=O)NCC2C3COCC23)CC12CCC2 73133,N1(C(=O)Nc2nnc(C)s2)CCn2ncc(Cl)c21 73134,c1(CC)ccccc1CC(=O)NCC(C)CN(C)C(C1CC1c1nccn1C)=O 73135,Cc1nc(CNC(c2nnnn2CCN2CCOCC2)C2CCOC2)cs1 73136,c1(C(C(=O)NC(CC)C)N(CC(C)C#N)C2CC2)ccc2nonc2c1 73137,n1(C(C)C)cc(C(N2CC3CC2C3CNC(=O)C(C)C2CC2)=O)c(O)nc1=O 73138,c1(C(N2CC(NC(=O)C3CC3)C(F)CC2)=O)ccc2oncc2c1 73139,N1(C(C2C(C)(C)C2(F)F)=O)CCCC2(C1)OCC(O)C2O 73140,C1(CN(C(=O)CSc2cnn(C)c2)CC)CCCCN1C(=O)C=Cc1ccco1 73141,N1(C(C#CCNC(C=C(C)C(C)C)=O)=O)C2CCC1CC(O)C2 73142,N1(C(C2(SC)CC2)=O)CC(CNC(=O)C(=Cc2ccccc2)OC)C2(CCC2)C1 73143,Cn1ncc(C(=O)NCc2csc(CNC(C3C=CC=CC=C3)=O)n2)c1F 73144,C(=O)(CC(O)CN(C)C)N1CCC(OCC)C1.C12(O)CC(C1)NC2=O 73145,C(C1CN(C(=O)C=Cc2ccoc2)CC1C(=O)NC(C)CN=[N+]=[N-])=CC 73146,c1(C(c2nnnn2C)NCC#CC)ccnc2[nH]c(C(F)F)nc12 73147,C1(CNC(Cc2cc(C)no2)=O)CCN(C(=O)CCCF)CC1O 73148,N1(C(Cc2nc(CC)sc2)=O)CCOC(C)(CNC(c2cc(C)cs2)=O)C1 73149,c1(COC)cc(C(=O)NCCCCN(C)C(C2CC2c2cncn2C)=O)no1 73150,Cc1ccc(O)c(CN2CCC(C)(C(=O)NCc3cc(F)cc(Br)c3)C2)c1 73151,c1(CC)[nH]c(Cl)nc(=NCC2(NC(c3ccncc3)=O)COC2)c1C#N 73152,c1(C(=O)NC(C)CCNC(=O)Cc2ccccc2CC#N)ccc(N=[N+]=[N-])cc1 73153,c1(CC)nc(O)c(C(=O)NCC2CN(C(=O)C(C)COC)C2)cc1C 73154,N1(C(C2CC(=C3CC3)C2)=O)CCC2OCCN(C(=O)Cc3ccc(F)cc3F)C2C1 73155,Cc1c(C(N2CCC(NC(=O)Cc3cncs3)C2)=O)nnn1C1CCOC1 73156,N1(CN=C2NCC(=O)N2)CCC(C2CCCN(C(=O)CC(F)(F)F)C2)C1 73157,Cc1ccc(OC(=O)C(Cc2ccccc2)OC(C)C)cc1I 73158,c1(OC)ccc(O)cc1CN1CCC(F)(C(N2CCC(C(F)F)CC2)=O)C1 73159,c1(C(N2CC(NC(=O)C=Cc3ncc[nH]3)C(C(F)F)C2)=O)c[nH]c2cccnc12 73160,N1(c2ccnc(COC)n2)CCC2CCN(C(C34CC3COC4(C)C)=O)CC2C1 73161,C1(CC)(CC)CC(NC(=O)CN=S(C)(C)=O)CN1C(c1ccc(N(C)C)nc1)=O 73162,N(S(=O)(=O)N1CCC2(CCCC2)CC1)C1CCN(CC(N)=O)CC1 73163,CC1(C)CCCN(C(=O)COCC(F)F)C1CNC(=O)COc1ccncc1 73164,c1(OC)ccc(CO)cc1O.C12CN(C(=O)CC3COC4CC3C4)CC1NC2=O 73165,c1(C(=O)NC(CC)CN(C(=O)C(C)(C)C(C)C)C)cccc([N+](=O)[O-])c1 73166,C(=O)(CC(=O)NCCOC(C)(C)CNC(=O)CCN(S(C)(=O)=O)C)N(C)C 73167,C1(C(=O)NC2CC(NC(CS(CC)(=O)=O)=O)C2)CCCC2(CCC2)C1 73168,c1(OCCNC(N2CC(C=C)OCC2)=O)cccc2ccccc12 73169,C1(N(C)C(C2CCCN2c2cnccn2)=O)CCCN(c2nccnc2F)C1 73170,c1(C(N(C(CNC(c2ccc(CCCCCC)s2)=O)C)C)=O)cnn2cc[nH]c12 73171,C(=O)(C(F)(F)C(C)O)NC(C(=O)NCc1nnn(CC)n1)CC1CC1 73172,c1(C(N(C2CCC2)Cc2cn(C(C)C(=O)O)nn2)=O)ccnc2ccncc12 73173,Cc1ccc2c(C(=O)NCCC3CCCN(C(C4(O)CCOC4)=O)C3)csc2c1 73174,C1(C(N(C2CCC(NC(C3CCNC3=O)=O)CC2)C)=O)CCC(C)(C)O1 73175,C(=O)(C(C)(C)C(=O)N1CC(CNC(c2cnc(C)[nH]2)=O)C2(CC2)C1)NC 73176,C(C(C(C)C(C)C)NC(c1cc(C)n(C)c1C)=O)NC(CCN(CC)CC)=O 73177,C1(C(=O)NC2CCC(C)(CNC(=O)C(F)(F)C3CC3)C2)(OCC)CCCCCC1 73178,C=C=C(C)CC(=O)N(CC(C)O)CCNC(c1cn(C)nc1CC)=O 73179,c1(CCC)[nH]nc(C(N2CC3C(NC(=O)C(C)C)C3C2)=O)c1[N+](=O)[O-] 73180,C=CCC(C)C(=O)NCC1(O)CC(CNC(=O)C=Cc2cc[nH]c2)C1 73181,C1(NC(C(n2c(C)cc(C)n2)C)=O)C2CCN(C(c3sccc3F)=O)C2C1(C)C 73182,N1(C(Cc2ccc(C)cc2)=O)CC2OCC(NC(c3coc(C(F)F)n3)=O)C2C1 73183,CCC(O)C(C)(C)C(=O)NCC(C)CNC(=O)CCCCN(C)C(C)C 73184,N1(C(C2(C)CN(C(c3sccc3I)=O)C2)=O)CCC(N2CCCC2)CC1 73185,C12CCCN(C1)C2=O.C(C(C)CN(C1CC(SC)C1)C)OC 73186,c1(OC)ccc(Cl)cc1S(=O)(=O)NC1CN(Cc2c[nH]c3c(F)cccc23)C1 73187,c1(CC(C(=O)N(CCC(C)NC(c2cnsc2)=O)C)=O)cccc(Cl)c1 73188,N1(C(C)=O)CCCC1CC(=O)N(CCCN(C(=O)CSCC1CCOC1)C)C 73189,N1(C(CCCC)=O)CC2CCCC2(C(=O)NC(C2CCCC2O)C)C1 73190,N1(C(C2=C(C)OCCS2)=O)CCCC2CN(C(C3(O)CCSCC3)=O)CCC12 73191,c1(C(=O)NCCCN(C(=O)CC(C)C)CC)cc(Cl)n[nH]1 73192,c1(CC(N2CCC(O)(CN(C(C(CC)SC)=O)C)C2)=O)ccc2cnccc2c1 73193,C1(C(=O)NCC(=O)OC23CC(F)C2C3)CC2(CCCC2)CO1 73194,C1(NC(C(C)OCCCC)=O)CCN(C(=O)Cc2cc[nH]c(=N)c2)CC1C 73195,CC(CN=c1[nH]c(=NC2COC(C3CC3)C2)[nH]c2ccc(Cl)cc12)C1CCCC1 73196,Cc1cnc(C(=O)NCC2CCCCN(C(=O)C=Cc3ncc(C)[nH]3)C2)c(F)c1 73197,C1(CC(=O)NCC2CN(C(C3CC34CCOC4)=O)C2)CCC=CCC1 73198,C1(C(N2CC3C(NC(C(=C(C)C4CC4)F)=O)C3C2)=O)COC2(CCC2)CO1 73199,CC1CCC(NC(C2(F)CCCC2)=O)CN1C(=O)C(=O)Cc1cccc(Cl)c1 73200,C1(CN(C)C(c2cc(F)n[nH]2)=O)CCCN1C(=O)CCc1nc[nH]n1 73201,c1(C(=O)NC(CN(C(C2CC2CC(C)C)=O)CC)C)c(Br)ccc(F)c1N 73202,c1(OC)ccc(C(=O)NCC(C2CCC2)NC(=O)Cc2cncc(C)c2)c(F)n1 73203,CC(C)CC(C)CC(=O)NCC1(F)CCC(NC(c2ccc(F)cc2)=O)C1 73204,C1(NC(Cc2ccc(OC)c(OC)c2)=O)CC12CCN(C(=O)C(C)(C)C#N)CC2 73205,c1(C(N2CCC(O)(CC#N)C2)C(=O)NCCCF)cc(I)ccc1F 73206,c1(CC(=O)NCCOCCC(=O)NCCCOC2CCC2)cccc(O)c1 73207,C12(CNC(=O)C(F)n3ccnc3)CCC(CC1)N(C(c1cc(F)cnc1O)=O)C2 73208,C1(C(N2CC(n3cc(CNC(CNC(C)=O)=O)nn3)C2)=O)CCCC(C)(C)CC1 73209,c1(CCC(=O)NCC(N2CCCC2CN(CC)CC)=O)c[nH]c2c(C)cccc12 73210,C(=O)(C1=COCCC1)NC1C(C(=O)NCCn2c(C)ncc2)CCOC1 73211,C12(NC(c3cccn4ncnc34)=O)CCCC1N(C(=O)C1=NOCC1)CC2 73212,N1(C(c2ccc(N)cc2F)=O)CC2CCC(C1)N2C(C1CCCC(F)(F)C1)=O 73213,c1(CC(=O)NCCC(C)NC(=O)C(C)(C)n2cnnn2)ccc2nn(C)cc2c1 73214,Cn1cncc1C=CC(=O)NC(C1CCCCC1)CNC(C1COC(=O)O1)=O 73215,N1(C(C(=O)Nc2cn(C(C)C)nc2)=O)CC(C(N)=O)C(C(F)(F)F)C1 73216,N1(c2snc(C(=O)OC)n2)CCC2(CCCN(C(=O)Cn3c(C)csc3=O)C2)C1 73217,c1(CNC(=O)NCC(N(OC)C)=O)cc(F)ccc1N(C)C1CC1 73218,N1(C(c2c(Br)cn(C)n2)C(=O)NC2(C)CC2)CCC(C(N)=O)(N(C)C)CC1 73219,N1(C(C(C)(C)OCCC)=O)C2CCC1CN(C(=O)CC(C)(O)COC)C2 73220,C(=O)(C1=NOC2COCC12)NCC(CC(=O)Nc1ccc(C)nc1C)O 73221,C#CC1(C(=O)NCc2ccccc2CC)CN(C(c2cn(C)cn2)=O)C1 73222,Cc1nc(C(=O)NCC2CCN(C(C3CCNC(=O)C3)=O)C2(C)C)ccc1C#N 73223,C1(NC(c2[nH]cc(C(C)(C)C)c2)=O)CCOC(C(=O)NCC=C2CCOCC2)C1 73224,c1(C(=O)NCC(CN(C(c2c(OC)c(Cl)sc2)=O)C)O)ccc(F)c2[nH]ccc12 73225,CC1CC(N(C(=O)C(=O)NCc2cccc(C(C)(C)C)c2)CCO)CCO1 73226,CCCC(C)(O)C(=O)NC1CCCC(NC(C2CC(F)(F)C2)=O)C1 73227,N12CCCC(C1)NC(=O)C(CC)N(CC)CC2=O.C1(CCOCC)(CSC)CC1 73228,C1(C(N2CC(C3(NC(CCN(CCC)C)=O)CC3)C2)=O)CC2OC(C)(C)OC2C1 73229,c1(C(N2CC(C(=O)OC)C(OC)CC2)=O)cnc(O)c2cccnc12 73230,N1(C(C(C)Cn2cccn2)=O)CC(NC(c2c(Cl)cnn2C2CCCC2)=O)C(O)C1 73231,c1(COCC)nc(-c2cc(Br)c(CC)s2)n(-c2ccnc(F)c2)n1 73232,C1(C)(C(=O)NC2C(NC(Cc3ccn(C)n3)=O)CC2)CCC12CCC2 73233,CC1(CNC(C2CC(NC(=O)CCN=[N+]=[N-])C2)=O)CCCCO1 73234,N1(C(c2cc(C)c(C)o2)=O)CCCCCC(Nc2ncc3ncn(C)c3n2)C1 73235,c1(C(CCC)C)nc(Cc2cc(C)n(C)n2)n(-c2cccc(Cl)c2)n1 73236,C1(O)(CNC(CNC(C(CC)C)=O)=O)CCCN(C(C23CC(CC)(C2)C3)=O)CC1 73237,Cc1cccc(C(C(=O)NCCCF)N(CCC(C)C)Cc2ccccc2)c1 73238,c1(CC(N2CCCN(C(C(C)NC(C)=O)=O)CC2)=O)coc2ccccc12 73239,c1(C(c2n(C(CC)(C)C)nnn2)NC2CC3(CC3)C2)cc(C)ncn1 73240,c1(C(=O)OCC)cnc(N2CCCC2CNC(=O)CC2CCCCO2)nc1 73241,C(=O)(CCCS(N)(=O)=O)NCCC(C)N(C(Cn1nc(C)n(C)c1=O)=O)C 73242,c1(C(N2CCC(C(C)NC(COCCC(C)C)=O)C2)=O)cccc2c1CNC2=O 73243,N1(C(c2cn(CC=C)nn2)=O)CCCCCC(NC(C2(COC)CCCC2)=O)C1 73244,C1(CC(=O)NCC2CCN(C(C3(NC(N)=O)CC3)=O)C2)(CC)CCCC1 73245,c1(CC(=O)NC(C2CCN(C(CCCNC(C)=O)=O)C2)C)ccc(Cl)cc1 73246,C1(C(N2CC(CC(C)NC(C3CCCCC3O)=O)C2)=O)C2CC3CC(C2)CC1C3 73247,C1(NC(c2c(CCC)occ2)=O)CC(C)CN(C(c2ccn(CCO)c2C)=O)C1 73248,N1(C(C2C3(CC(OCC)C3)C2)=O)CC2CC(NC(=O)C(=O)C(C)(C)C)C1C2 73249,CC(C)(CC(F)C(=O)NCC1CNC(=O)O1)NC(=O)CCC1CCC(=O)C1 73250,c1(C(N2CCN(C(=O)CC3CCCCC3)C(CO)C2)=O)cc2ccc(Cl)nc2s1 73251,c1(N(C(c2cnn(C)c2)C)C(C2CCNCC2)=O)ncncc1Br 73252,c1(-c2nc(-c3c(C)scn3)n(CCC(=O)OC(C)(C)C)n2)ccc(OC)c(Cl)c1 73253,CCC(CC)(CC)C(=O)NCC(C(C)C(C)C)NC(c1ccc(S(N)(=O)=O)s1)=O 73254,c1(OC)ccc(C(=O)Nc2ccc(C(=O)C(F)(F)F)cc2)c(O)c1F 73255,c1(SC)nc(N2CC(F)(C(=O)Nc3cc(I)ccc3F)C2)ncc1Br 73256,c1(C(C)C)sc(Cl)nc1C(N1CC(NC(=O)C(C2CCOCC2)O)C1)=O 73257,C(CNC(=O)CC1CC2(CC2)CO1)(CC(=O)N(C)C(C1CCCC1)C)OC 73258,C1(C)(NC(CC(C)(CNC(=O)COCCCF)OC)=O)CCC(C)C1 73259,CC(CC(F)(F)F)C(=O)N1CC(CC(=O)NCCC2CC2)CC1(C)C 73260,c1(C(=O)OC)c[nH]nc1S(=O)(=O)NC(CCSC)C(=O)OC(C)C 73261,N1(C(CN(C(C(CC)OCC)=O)CCOC)=O)CCCC(C(=O)OC)C1 73262,c1(C(=O)NC(C)CCCCNC(c2ccon2)=O)c(Cl)oc2ccccc12 73263,c1(OC)ncnc(C(=O)NCC2CCCCC2NC(=O)Cn2cnnc2O)c1F 73264,C(=O)(C(CO)C(C)(C)C)NCC1(C)OCCN(C(c2cnc(C(C)(C)C)[nH]2)=O)C1 73265,N1(C(c2nc(C(C)OCC)sc2)=O)CCC(C)(NC(=O)CS(=O)CC)CC1 73266,N#CCCCCCC(=O)NCCC1CN(C(=O)Cn2cc(CO)nn2)CCCO1 73267,c1(C(=O)NC2CN(C(c3ccc(C)cn3)=O)C(C)C2)cc(C(F)(F)F)ccc1O 73268,CC1CCCC(C(=O)NC(c2ccc(Br)cc2)(C)C(=O)O)O1 73269,c1(C(N2C(CCNC(C3CC(CC)C3)=O)CCC2)=O)ccc(N)c(F)c1Br 73270,c1(OC(C(N2CC(NC(C(C=CC)O)=O)C2)=O)C)cc(Cl)cc(Cl)c1 73271,Cc1cccc(C(C)C(=O)NC2CC2NC(c2cnn(C3CCC3)c2)=O)c1 73272,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1(CO)CN(c2c(OC)c(C)ncn2)C1 73273,c1(NC(C2CC(O)(CNC(c3cscc3C3CC3)=O)C2)=O)ccc(CCO)cc1 73274,N1(C(=O)C(C2CCCCC2)O)CCN(C(c2ccn3cccc3c2)=O)C2(CC2)C1 73275,C#CC(CNC(=O)CCCCNC(C1(O)CCOC1)=O)C(C)C 73276,c1(C(=O)NC(CCCNC(COCCOCC#C)=O)C)ncnc2cc[nH]c12 73277,C1(CNC(C=C(C)C(C)C)=O)CCCCN1C(C1CN(C(=O)OC(C)(C)C)C1)=O 73278,C(=O)(C1CCCc2scnc21)NCC1N(C(c2c(C)[nH]c(=NCC)s2)=O)CC=C1 73279,CC1COCC(C(=O)NC2CCC(C(N3CCC(c4cnco4)C3)=O)CC2)O1 73280,CCCC(C)CCCC(=O)NCC1(F)CCCN(C(=O)Cc2ccno2)C1 73281,C(=O)(C(C#N)(CC)CC)NC1CCC(NC(C(CC)N(CC)CC)=O)CC1 73282,c1(C(N2CCN(C(c3c(C)nn[nH]3)=O)CC2C#N)=O)cc2cc[nH]c2cc1F 73283,C1(NC(C(C)=CC2CC2)=O)CCCC(NC(c2c(C)noc2C(C)C)=O)C1 73284,C1(CNC(=O)CCCc2cnccn2)C(F)(F)C12CC2 73285,c1(NC(CC=C)C)[nH]c(=NCc2cnc[nH]2)nc2c1ncn2C 73286,O=S(=O)(c1nccs1)Nc1cccnc1.C12(F)CCN(CC1)C2 73287,C1(NC(c2cc(CNC(=O)C(F)CC3CCOC3)cs2)=O)CCC2(CC2)C1 73288,C(CC(CNC(c1cc(C)co1)=O)NC(=O)C=CC1CCCO1)OC 73289,CCCCC(CC)C(C(=O)NC1CCCCC1)N1CCCCC1c1ccco1 73290,C1(C(=O)Nc2ccc(C(C)C)cc2)CN(C)CCN1C(=O)C(F)C(F)(F)F 73291,C(=O)(C1=NOC(CNC(=O)Cn2ccnn2)C1)N1CCC(C)(N(C)CC)C1 73292,c1(C(=O)NCC(CC(N2CCCC(CC)C2)=O)O)n[nH]cc1[N+](=O)[O-] 73293,C(=O)(C1=CS(=O)CCC1)NCC12CC(NC(CC(=O)N(C)C)=O)(C1)C2 73294,CCC(C)C(C(=O)NCC(C)(C)CCOC)NC(c1ccccc1NC)=O 73295,c1(C(c2n(CC=C)nnn2)NCc2ccc(N(C)C)cn2)cccc2c1CCC2 73296,N1(C(C(C)N(C(C)=O)C)=O)CCC(C2CCN(C(C3(F)CCCC3)=O)CC2)CC1 73297,N1(C(C(C)(C)SC)=O)CCCN(C(=O)Cc2ncc(Cl)s2)C(C)C1 73298,CCC(C(=O)NCC1(F)CCN(C(c2cc(OC)n[nH]2)=O)CC1)C(C)O 73299,C1(C(=O)NC(c2nc(CC3CCCO3)on2)(C)C)CCCCN1S(C)(=O)=O.SC 73300,CC(C)(C)CCCN=c1ccc(S(=O)(=O)NCCCCC2CCCC2)c[nH]1 73301,c1(C(=O)NC)c(C)nc2cc(O)nn2c1C.C1(C)C(=O)N1CCCNC(CC)=O 73302,CCC(C(=O)N(CC(C)(C)CNC(=O)C(Cc1ccsc1)NC=O)C)C(C)C 73303,c1(OC)cc(C(=O)NC2(CO)CN(C(=O)C(O)CF)C2)cc(Cl)c1 73304,C(=O)(C#CC(C)(C)C)NCC1C(C(N2CCC(CCC#C)CC2)=O)C1 73305,c1(C(N2C(C)CC(CNC(c3n[nH]c(C)c3N)=O)C2)=O)cnn2c1CCCC2 73306,C(C)(CNC(=O)C(C)SCC)(CC(C)C)NC(CCC=C)=O 73307,C(=O)(CC(C)(C)C)NC(CNC(c1c(-c2ccn(C)n2)n[nH]c1)=O)(C)C1CCC1 73308,c1(OC)ccc(O)c(C(=O)NC2CCN(C(c3ccc(NC(C)C)cn3)=O)C2)c1 73309,N1(C(=O)OCC=C)CCN(C(=O)CCn2cc(C3CCCC3O)nn2)CC1 73310,C(=O)(C(C)CS(C)(=O)=O)NCC1CCCCN(C(CCCc2ccc(C)s2)=O)C1 73311,N1(C(CCNC(C)=O)=O)CCC(NC(=O)CS(=O)(=O)NC(C)(C)C)CC1C1CC1 73312,C1(NCc2c(C)c(C(F)(F)F)n[nH]2)CC2(CCC2)C12CCC2 73313,S(=O)(=O)(c1ccc(NC2COC3(CCCCC3)C2)nc1)NC(C)CCO 73314,N1(C(CCC2(NC(c3cncc(O)c3)=O)CCC2)=O)CC2C(CO)C2C1 73315,C1(CNC(C2CC(SC)C2)=O)COCCN(C(c2ccccn2)=O)C1 73316,c1(C(N(CC(C)NC(c2cnc(C3CC3)s2)=O)CC)=O)ccc2ncn(C)c2n1 73317,C12(C(N3CCN(C(C)C)CC3)=O)CCN(C(=O)CNC(N)=O)CCC1C2 73318,c1(C(=O)NCCC(=O)NCC)n[nH]cc1CNC(=O)COCC1CC1 73319,C=CCC(CC(=O)NCC(O)C1(Cl)CC1)NC(=O)C=C1CCC1 73320,c1(OC)ccc(NC(C2CC(F)(F)CN2Cc2scnc2C)=O)c(Cl)n1 73321,C(=O)(C(O)C(C)C)NCCC(C)NC(C(CC)c1ccccc1)=O 73322,N1(CC(N2CC(CN(C(C(C)SC(F)(F)F)=O)C)C2)=O)CCCC(N(C)C)C1 73323,C(C(=O)N(C)CCN(C)C(C1(Cl)CC1(C)C)=O)(C(C)C)n1cc(C)nc1 73324,c1(C(CNC(C23CC(C)C2C3)=O)NC(=O)Cc2nnc(O)s2)cccc(Cl)c1 73325,CC(CC(C)(C)O)C(=O)NC(c1cn(C(c2ccc(Cl)c(F)c2)C)nn1)(C)C 73326,c1(NC(CC)C)ccc(S(=O)(=O)NCc2nnnn2-c2cn[nH]c2)cc1Br 73327,c1(C(=O)OC)cc(NC(=O)C(F)(F)C(O)c2ccccc2)n2ccccc12 73328,CCC(C(O)C(C)C)NC(c1ccc(NC(=O)NCC2CC2)cc1)=O 73329,CCCCCCCCCCCCNC(c1ccc(OCC(=O)O)cc1)=O 73330,C1(NC(C2(CC)CC2)=O)CN(C(c2cccc(OC)n2)=O)CC2CCCC12 73331,N1(C(c2ccc(NC(C)=O)s2)=O)CCC(C)(C)C1CNC(C1CC(=O)N(C)C1)=O 73332,c1(C(N2CCC(NC(C3CCC(=O)N3)=O)C2)=O)ncc(F)cc1F 73333,C12(C(N3CCC(NC(CNS(NC)(=O)=O)=O)C3)=O)CCC(=O)N1CCS2 73334,c1(C(=O)NCCN(CC(C)O)C(c2cc(C(F)F)no2)=O)c[nH]cc1C(C)(C)C 73335,C(=O)(C(C)CC(F)(F)F)NC1CCC(C(=O)NCc2onc(NC)n2)C1 73336,CC1(C)CCCC(O)(CNC(=O)Nc2ccc3ccoc3c2)C1 73337,CC1CCN(CC(=O)NCc2ccccc2CNC(C2(C)CCC(C)C2)=O)CC1 73338,C1(CCC(=O)NC(C)C(C)NC(C2CC(OC3CC3)C2)=O)CCCOC1 73339,N1(C(C(C)CC(F)F)=O)CCC2C(CCCN2C(C2(O)CCCCC2)=O)C1 73340,c1(CNC(NC(COC)C)=NCC2CN(C)CCO2)nc2c(s1)CCC2 73341,N1(C(c2cc(CC)oc2C)=O)CC2CCC2(CNC(C2CCCCCC2)=O)C1 73342,c1(C(CCC)C)cn(CC(=O)OC(F)F)nn1 73343,CCS(=O)(=O)CC(C)N(C(C(=O)Nc1nc(C)c(C)s1)c1csnn1)C 73344,C1(NC(C(c2cc(C)oc2C)C)=O)CC2CN(C(=O)CCc3cn[nH]c3)CC2C1 73345,C(CCCC(=O)NC1(CO)CN(C(C2CCC(C#N)C2)=O)C1)NC(C)=O 73346,C1(C(N2CC(NC(C3(C)CCCC3)=O)C2)=O)CCC(N=[N+]=[N-])C1 73347,CN1C(=O)Cc2c(C(=O)NCC3C4CN(C(=O)Cn5cnnn5)CC34)cccc21 73348,c1(N2CC(NC(c3c(C)cn(C)c3)=O)C(C)(C)C2)c(F)cccc1[N+](=O)[O-] 73349,C(=O)(C(C)CCC(C)(C)C)NCC1(F)CCN(C(C(C)NC(CC)=O)=O)C1 73350,C1(CC=C)CCCCN1C(c1cn(CC)nn1)C(=O)NC(C)(C)CC 73351,C1(CC(N2CC(NC(CC=C(C)C)=O)C(n3cccn3)C2)=O)CCCNC(=O)C1 73352,C1(N(C(C2CCN(CC(C)C)C2)=O)C)CN(C(=O)CCc2ccco2)CC12CC2 73353,C1(C(=O)NC2CCCC(O)C2)CN(C(c2ccnn2C2CC2)=O)CC1(F)F 73354,N1(C(C2(COC)CC2)=O)CCC(OCC(=O)NCC2(C)CCCS2)C1 73355,c12ccc(cc1)[nH]2.c1(C(=O)NC2(CC)CC2)c[nH]nc1F.C12CC(C1)C(=O)NC2 73356,N(C1CCCc2c[nH]nc21)C(c1nccc(CNC(=O)Cc2cc[nH]n2)c1)=O 73357,c1(C(=O)OCc2c(OCC)cccc2)cc(S(N)(=O)=O)c(C)cc1C 73358,N1(C(C(CC)CC)=O)CCC(C2(CNC(=O)C3CC3)CCOCC2)CC1 73359,N12CCc3sccc3C1CNC(=O)C(F)(F)C(C1CC1)C2=O.N1(C2CC2)CCCC1 73360,C1(C(N2CCC(C(F)(F)F)(OC)C2)=O)CCN(C)CC1C(F)(F)F 73361,CC(C)CCC(CO)NC(C1CC(CNC(c2coc(CO)c2)=O)C1)=O 73362,N1(C(c2c(C)nsc2C)=O)CCC(C)C(CC(N2CCCCC2CCO)=O)C1 73363,C1(NC(CCN2C(C)(CC(C)C)CCC2)=O)CCC(F)(F)CC1 73364,C(=O)(C(C(C)(C)C)c1cc[nH]n1)N(CCN(C(=O)CCOCC1CC1)C)C 73365,c12ccn(n1)CC(C)N2.CCS(=O)(=O)N1CC(C(=O)CNC(=O)OC(C)(C)C)C1 73366,CC(C(=O)NNC(=O)OC(=O)Cn1nnc(-c2ccsc2)n1)N(C)CC(C)(C)C 73367,N1(C(c2c(CC)noc2)=O)CCCC(C2CCN(CCOC3CCCC3)C2)C1 73368,C(C1=NOC2CN(C(C3(C4CC4)CCOCC3)=O)CC12)NC(c1cccnn1)=O 73369,C(C(C)(O)C(=O)N1CCC(NC(=O)Cc2ccc(CO)cc2)C1)OC 73370,C(=O)(C1=CCCCCC1)N(C(C)C(=O)Nc1cc(Cl)cnc1C)CC 73371,C=CC1(NC(C23CC2CN(C(C2CCC(O)C2)=O)C3)=O)CCCC1 73372,N1(C(C=C2CCN(C)C2)=O)CCC(NC(=O)CC2(C)CC(F)(F)C2)C(O)C1 73373,c1(C(N(CCCNC(C2(C=C)CCCCC2)=O)CCO)=O)cn2cccnc2n1 73374,c1(C(=O)NC2CCC(NC(=O)C=CC3CC3)C2)cc2ccncc2o1 73375,CC(C(=O)NC1(C)CCCN(C(c2cccc(Cl)c2F)=O)C1)C(C)(F)F 73376,C(CCCCC(=O)NC1(C(=O)NOCC2(C)CC2)CCCCC1)NC(C)=O 73377,Cc1nc(S(C)(=O)=O)sc1C(=O)OCC1CC(C(=O)OC(C)(C)C)C1 73378,C1(NC(C(C)NC(C)=O)=O)CC(F)CN(C(=O)C(C(C)C)c2cccc(Cl)c2)C1 73379,S(=O)(=O)(c1ccc(NCCc2ccnc(Cl)c2)cc1Cl)NC(CC)CO 73380,c1(CC(=O)N(CCCNC(c2cn(C)c(=O)n2C)=O)C2CC2)ccc2ncsc2c1 73381,CN1C(=O)CC(C(N2CCC(CO)C(NC(C3C4(CC4)C34CC4)=O)C2)=O)NC1=O 73382,c1(OC)ncc(C)cc1-c1ccc(C(C)NC(=O)Nc2ccccn2)nc1 73383,N#Cc1cc(Br)ccc1CN1CC2(CC2C(N2CC(O)CC2C(N)=O)=O)C1 73384,C1(C(N2CC(CC)N(C(=O)C=CC3CCOC3)CC2)=O)CC(F)(F)CCC1(C)C 73385,c1(OC)ccccc1NCC(=O)NCC1(O)CN(C(c2nc(Br)c[nH]2)=O)C1 73386,c1(N2CCC(NC(C)=O)C2)ccc(S(=O)(=O)NCCC2COC(C)(C)C2)cn1 73387,C1(C(=O)NC(CC)(C)C(=O)Nc2ccc(SC)cc2)CCc2ccccc2N1 73388,CCC(C(=O)NC1CCCC1NC(=O)C=CC(=O)N(C)C)n1ccnc1 73389,CC(C)CC(C(=O)NCC1(C)CCN(C(=O)CC2C=CCC2)C1)C(N)=O 73390,C(=O)(C(CC(C)C)N(C)C)NCc1c(CCNC(CC(=O)NCC#C)=O)ocn1 73391,C=C(C)CCCC(=O)NCC1COCC1NC(=O)C(C)NC(C)=O 73392,c1(N2CC=CC(N(C)C(c3cnc4sccc4c3)=O)C2)ncnc2c1nnn2C 73393,C12(NC(c3csc(C)c3C)=O)CCC(CC1n1cc(C3CC3CO)nn1)C2 73394,CCCC(CC(C)C)C(=O)NCc1ncccc1C(=O)N(C1CC(C)(C)C1)C 73395,Clc1cc(-c2nc(C3CC3)nn2CC2CC2)ncc1Br 73396,C1(C(N(C2C3CN(CC(F)(F)F)CC23)C)=O)CCCN(C(N)=O)C1.C12CN(C1)C2 73397,C1(CC(=O)NCC(C)(Cn2cccn2)NC(c2cc(F)n[nH]2)=O)NC(=O)NC1=O 73398,C1(NC(C=CC=CCC)=O)CCC12CN(C(=O)CC(c1ccc(F)cc1)C)C2 73399,N1(C(CCc2onc(CC)n2)=O)CC2CC(C1)N(C(=O)CCC1CCC(=O)N1)C2 73400,C(C(=O)N(C)CC1CCN(C(c2ccnc(S)c2)=O)C1)(C(C)C)c1cc(C)no1 73401,CC(CC(N)=O)C(=O)NCCOC1CCN(C(c2nc(C3CC3)ncc2Cl)=O)C1 73402,Cc1cc(Cl)c(C(=O)NCCN(C(=O)CCC2CCC(C)O2)C2CC2)cn1 73403,N1(C(CN(C(C(CC=CC)C)=O)C(C)C)=O)CC2(CNC(=O)OC2)C1 73404,C1(N(C)C)CC(N=c2ccnc(N3CCCC(c4nncs4)C3)[nH]2)C1 73405,c1(-n2cc(CC3(O)CN(C(=O)CCOCC(F)F)C3)nn2)cccc(F)c1F 73406,C(C(=O)Nc1ccccc1)(C1=CCC2CC1C2(C)C)N1CCC(S(CC)(=O)=O)C1 73407,C1(CNC(C2C(C)C2(F)F)=O)CC2(CCC2)CN1C(c1ccn(C)c1)=O 73408,Cc1c(F)c(F)c(C(=O)NCC2CCC(C)C2)c(F)c1F 73409,N1(c2snc(C(C)(C)C)n2)CCC(NC(C2CCCN(C(=O)C3CC3)C2)=O)C(F)C1 73410,CC1N(C(=O)N(CCCCC2CC2C)CCO)CCOC1(C)C 73411,C(CCCC)(C(=O)NC1(CCC=C)CCC1)NC(COCCCC#C)=O 73412,Cc1nc(O)nc(C)c1C(=O)NCCC(C)NC(=O)Cc1cnn(C(C)(C)C)c1 73413,c1(N2CCN(OCC)CC2)n[nH]c2ccccc12 73414,Cc1c(C(N2CCN(C(C3CC34CCC4)=O)CC2C(C)C)=O)cnc2nncn12 73415,CCCC(C)C(=O)NC1(CCC(=O)NCc2cn(C)nc2CC)CCCC1 73416,c1(OC)cc(C#N)ccc1N(C1CC2CNC1C2)C(=O)CCc1cnc[nH]1 73417,C1(C(=O)NCCC(C)NC(C2(C)CCSCC2)=O)CCOC(=O)N1 73418,N1(C(c2c(C)cc(C)s2)C(=O)NC(C)C)CCCC(C)(O)C1 73419,c1(NC(=O)NC(C=C)C2CCC2)ccc(OC(F)F)c(F)c1 73420,N1(C(C(C2CCOC2)OCC)=O)CCN(C(C2CC(C)CCO2)=O)CC1CCO 73421,CC1(C)CCCN(C(c2cc(N)cc(O)c2)=O)C1CNC(=O)CNc1nccs1 73422,C(=O)(C(C)(C)CCC(=O)OC)N1CCN(CCN(C(CCCC(=C)C)=O)C)CC1 73423,c1(C(C(=O)NC(CCN(C(CC=C(C)C)=O)C)C)O)ccc(Cl)cc1 73424,c1(C(N2CCC(N(C(c3ccc(F)c(Cl)c3)=O)CC)C2)=O)ccc2c(c1)CCO2 73425,C1(C(=O)NC2C(NC(=O)Cc3cscn3)CCC2)CCC12CCC2 73426,c1(OCC(=O)NCC2CCCCN2C(c2csc(C(F)F)n2)=O)ccc(F)nc1 73427,C1(C#N)(SC)CN(C(=O)C(Cc2ccoc2)NC(=O)CC2CC(N(C)C)C2)C1 73428,C(=O)(CC(O)C(Cl)(Cl)Cl)NC1CC(C)(NC(c2cc(CCO)on2)=O)C1 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73621,C1(NC(C(N2CCCC(C)C2)=O)=O)CCC12CN(C(c1ccncc1)=O)C2 73622,N1(C(c2nn(C)c(Br)c2C)C(=O)NCCOCC)CCN2C(=O)NC(=O)C2C1 73623,C(N=c1cc(NCCC2=CCCCC2)nc[nH]1)c1ncn(C)n1 73624,c1(N2CCC(C(=O)NC(CCC)Cc3nccn3C)C2)ccc2c(c1)OCO2 73625,CC1(C)CCC(CNC(c2ncc3ccccn23)=O)N(C(C2C=CCCC2)=O)C1 73626,CCC(C)(CO)C(=O)N1CCOC(CCCNC(=O)C(F)=CC2CC2)C1 73627,c1(-n2c(Cn3ccc(C(F)F)n3)nc(COC(C)C)n2)ccc2ncsc2c1 73628,N1(C(C2C(OC)CCC2)=O)CCCC(C)(C)C1CNC(=O)CCC1CC1 73629,C(=O)(CN=S(C)(=O)c1ccc(Cl)cc1)NC1(C)CCCC1NC(=O)C(F)(F)F 73630,c1(OC)ccc(OC)c(S(=O)(=O)NCCCNCC)c1.c1(C2C(N)C2)cccs1 73631,Cc1cc(NC(C2(C)CCCN2C(=O)Cn2nccn2)=O)cc(O)c1 73632,C(CCCC(C)NC(C1CCOCC1)=O)NC(c1nc(C(=O)OCC)sc1)=O 73633,c1(SC2CCN(C(=O)CN3CC4C(CO)C4C3)CC2)c(Br)ccc2c1OCO2 73634,N1(C(c2cc(O)ncn2)=O)CC2COCC2C1 73635,C1(C(N2CC(CC(C)NC(=O)CCSCC(N)=O)C2)=O)(OC)CCOCC1 73636,c1(C(C)C)ccc(C=CC(=O)NCCN(C(c2ccccc2)=O)C(C)C)cc1 73637,N1(C(C2(F)CCN(C(c3ccc(NC=O)cc3)=O)C2)=O)CCc2n[nH]cc2C1 73638,C(=O)(C1=CS(=O)(=O)CCC1)NC(C1(O)CCN(C(c2ccn(CF)n2)=O)CC1)C 73639,N1(C(c2c(C)coc2)=O)CCN(C(=O)C(F)(F)Oc2ccccc2)C(C)C1 73640,c1(C(=O)NCC2C(NC(CCn3ccc(C)n3)=O)COC2)ccn2nncc2c1 73641,Cc1nc(-c2cn(CCCCNC(=O)Cc3nc(C(=O)O)co3)nn2)cs1 73642,N1(C(CC(C)OC)=O)CCC(C)C1C(=O)NCCc1ccc(C)nc1 73643,C12CCC(CC1)C(=O)N(C(C)(C)C)C2=O.C(C)(CC(=O)OCCN)SC 73644,CC1=C(C(=O)N2CC3(C2)CN(C(=O)C(F)CC=O)C3)C(C)(C)CCC1 73645,C(c1c(C)coc1C)=CC(N1C(CCNC(CC2N(CC)CCC2)=O)CCC1)=O 73646,C1(C(=O)NC2CC(CC)(CC)C2)CC(F)(F)CN1C(=O)CC1COCC(C)O1 73647,C(=O)(C(C#N)=CC1CC1)N(C1CC(NC(=O)CC2(C)CC2(Cl)Cl)C1)C 73648,C=CCCCCCCC(=O)NC1(CNC(c2cncc(C)c2Cl)=O)CCOCC1 73649,N1(C(C2N(C(C3CC4(CC(C)C4)C3)=O)CC2)=O)CC(O)C(O)C12CCC2 73650,N1(C(C(c2ccnn2C)NC(C(C)C#N)=O)=O)CCCCCCCCC1 73651,CC(C)CC(=O)NC1CC(N(C(=O)CC2CC(C(F)F)C2)C)C1 73652,Cn1cncc1CC(N1CC(CCCCNC(=O)CCCn2cccn2)C1)=O 73653,C1(Cn2cc(C(CC)(C)C)nn2)CC(O)CN1C(c1coc(C)n1)=O 73654,O=C(C1=CCCOC1)NC1(CO)CCN(C(c2ccccc2)=O)C1 73655,Cc1cc(C(N2CC3CC(NC(C4CC45CCC5)=O)C2C3)=O)ccc1C(F)(F)F 73656,C(=O)(C(CC(F)F)NC(=O)CCCF)NCc1n(CC)cnn1 73657,Cc1nc(C(=O)NCc2c[nH]nc2C(=O)NC2CCC2O)c(C)s1 73658,c1(OCCC(=O)NCC(C(C)C)NC(C2(CC)CCCO2)=O)ccccc1OC 73659,C=CC(C)C(C)C(=O)NC1(C)CC(NC(c2cncc(Cl)c2Cl)=O)C1 73660,CCCCCCC(C)CC(=O)NCC1CCN(C(=O)C(C)(C)C2=CCSCC2)C1 73661,C1(C(C)C)CNC(=O)CN1C(=O)CCCCCn1cc(-c2cccnc2)nn1 73662,C(=O)(C(C)(C=C)CC)NCc1cncc(C(=O)NC(C=C)(C)CC)c1 73663,CN1CCC(C(=O)NCc2ncoc2C2CN(C(=O)C(=O)NCC(F)F)C2)C1 73664,Cc1ccc2oc(C(N3CC4(CCCN4Cc4cccc(C)c4F)C3)=O)cc2n1 73665,CCCC(C(=O)NCCC(O)C(=O)N(CC(F)F)CCC)C(C)C 73666,C1(CC(N2CCC(C(=O)NC)C2)=O)CC(C)(C)CCO1 73667,CC1(NC(C2CCCS2)=O)CC(NC(c2cnoc2C2CCC2)=O)C1 73668,C1(N(C(c2c(C)ocn2)C(=O)NC(C)C)C)CC(O)C1(C)C 73669,C1(C)(C(=O)NCCCCC(C)NC(C2(C)CC3CCC2C3)=O)CC2CCC1C2 73670,CC1(C(=O)NCC2(C)CCN(C(=O)Cc3csc(Cl)n3)C2)COC(=O)OC1 73671,C1(COC)(NC(=O)Cc2ccccc2Cl)CCN(C(=O)C(F)OC(F)(F)F)CC1 73672,c1(COC(=O)CC(c2ccccc2)n2cccc2)ccc(I)c(Cl)c1 73673,C(CCF)(C(=O)N1CC(C(C)O)C1)NC(COCCC#C)=O 73674,c1(CNC(C2CC2Nc2cc(OC(F)F)ccn2)=O)cccc(I)c1 73675,C1(CCNC(=O)CN2CCOCC2)CCN(C(c2csc(CO)n2)=O)CC1(F)F 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73694,C1(CC)(CC)CN(C(=O)C(C)(C)C(C)NC(=O)COCC(=O)OC)CCO1 73695,C(=O)(C(O)(C(F)(F)F)C1CC1)N1CC2C(CNC(Cc3nnc(C)s3)=O)C2C1 73696,N1(c2nnc(-c3[nH]n(C)c(=O)n3)n2C(C2CCCCN2C2=CC=C(Cl)CC2)=O)CCC(F)(F)C(F)C1 73697,c1(OC)ccc(C(=O)NC2COCC2NC(C2(C(F)(F)F)CC2)=O)nn1 73698,C1(C(N(C2CCN(C(c3cn(CCO)nn3)=O)C2)C)=O)CC(=O)NC(=O)C1 73699,c1(C2(N(C(CN(C(CCC)=O)C)=O)C)CC2)nnc(O)n1C.C(C(=O)OC(C)=O)=C 73700,CC(C)(N=[N+]=[N-])C(=O)NCC1(CNC(=O)CNC=O)CC1 73701,C1(NC(c2c(OC)n[nH]c2)=O)CN(C(=O)C(N2CCCC2)C2CC2)C2(CCC2)C1 73702,c1(C(=O)OCC)c(NC(C2CC(F)CN2C(=O)C2=CCCS2)=O)cccc1C 73703,CC1(CO)C=CCN1C(=O)CCOCCNC(c1cccc(O)c1)=O 73704,C(=O)(C(C)C(=O)NCc1cc(C(N2CCCC2(C)CC2CC2)=O)n(C)n1)OC 73705,C(CC(C)(C)C(=O)NCCC1(CO)CCC1)NC(C(CCSC)O)=O 73706,CN1CCN(C(C2(CNC(=O)CCCN3CCCC3)CC=CC2)=O)CC1 73707,C1(C(=O)NC2CC(C(=O)NCC(=O)NC3CCC3)C2)(CC)CCCC1O 73708,c1(C(N2CCC(NC(CCc3cccc(OC)n3)=O)C2C)=O)cc(C)c(O)nn1 73709,N1(C(CC2OCC(C)(C)C2)=O)CCC2CN(C(C3CS(=O)(=O)C3)=O)CCC12 73710,c1(CC)c(OC)cccc1C(=O)NC(C)C(C1CCCCC1)O 73711,c1(SCCC(=O)NC)ccc(-c2cn(-c3ccccc3C(=O)O)nn2)cc1 73712,c1(CN(C)C)cccc(C(N2CC=CC2CNC(c2cccc(Cl)c2)=O)=O)c1 73713,N1(C(C2CN(C(CN3CCC(NC(C)=O)CC3)=O)C2)=O)CCC2OCCCC2C1 73714,Cc1cc(COCC(=O)NCC(C)CN(C(=O)CC2CC=CC2)C)no1 73715,c1(C(=O)NCC2N(C(CC(n3ccc(C)n3)C)=O)CC=C2)oc(C(F)F)cc1C 73716,C1(O)(CNC(C2CC2CF)=O)CCN(C(=O)CCC=CBr)CC1 73717,Cc1cc(C(N2CC3C(CNC(C4(C)CCN(C)C4=O)=O)C3C2)=O)cc(C)c1 73718,C1(OC)CN(c2cc[nH]c(=N)n2)CC1NC(=O)NC(C)C 73719,CC(=O)CCCC(C)C(=O)NC1CCN(C(=O)C(=C2CCCCC2)F)C(C)C1 73720,C1(C(N(C2CCN(C(C3(C)CC=CC3)=O)C2)CC)=O)COCC1(C)C 73721,c1(C(=O)NC2C3CCC2N(C(c2occc2F)=O)C3)cc2ccc(F)cc2o1 73722,Cc1cc(CC(=O)NCCC2(O)CN(C(=O)CCc3ccc(C)s3)C2)on1 73723,N1(C(C(c2ncc(C)s2)C)=O)CC(O)CC1CC1CCNCC1 73724,c1(C(N2C(CN(C(CNC(=O)OC)=O)C)CCC2)=O)cc(Cl)cc(F)c1F 73725,c1(C(=O)NCC2CCN(C(C(CC=C)CC)=O)C23CC3)cc2ccccc2cn1 73726,C1(CC(=O)NCCc2ccns2)CN(C(=O)C=Cc2cc[nH]n2)CC12CC2 73727,C1(CNC(=O)COCC2CCCCO2)CCCN(C(=O)Cc2nnc(O)s2)CC1 73728,c1(C(N(CC(CNC(c2c(C(C)C)occ2)=O)C)C)=O)cnc2[nH]ncc2c1 73729,N1(C(C2(Br)C(C)(C)C2)=O)CCN(C(=O)CCCn2cccc2)CC(O)C1 73730,c1(CC(C)C)cc(N2CC3C(CNC(=O)C(C)Cn4ccnc4)C3C2)ncn1 73731,c1(CC(C(=O)NCC2(O)CN(C(C3(OC)CCC3)=O)C2)O)cc(Cl)sc1Cl 73732,C1(C(=O)NCCCN(C(c2cccc(C)c2O)=O)CC)CC12CCC(F)(F)CC2 73733,O=C1CC(C(=O)OC(C(=O)NCc2cccc(Br)c2)C(F)(F)F)C2(CCC2)C1 73734,c1(C(=O)NCC(CO)NC(c2ccc(CO)o2)=O)cc2ccc(Cl)cc2[nH]1 73735,C(=O)(C(F)CC(C)C)N(C1CCCN(C(c2n(CC)ccc2)=O)C1)C 73736,C1(CNC(C(C)(C)OCC)=O)CC2CN(C(C3CCC(C(N)=O)C3)=O)CC12 73737,C1(C)(COC)CCN(C(C2(CO)CCN(C(C3CCCCO3)=O)C2)=O)CC1 73738,C(=O)(CCCCCCCC)N1CC(CNC(C(CC#C)(C)CC)=O)C(C)(C)C1 73739,C12(C(=O)NCC3N(C(COCC)=O)CCC3)CCOC1CCOC2 73740,N1(C(C(F)=CC)=O)CCOC2(CCN(C(c3cscn3)=O)C2)C1 73741,C1(NC(C(CCC)N(C)C)=O)CC12CCN(C(c1ccc(CC)s1)=O)CC2 73742,C12CCCN(C1C)C2.c1(-c2cc(OCC)ncc2)cc(F)cnc1OC 73743,N#CC1(C(=O)NCCC2CCCN(C(c3ccncn3)=O)C2)CCOC1 73744,c1(OC)c(C(=O)NC2CC(CNC(=O)C(C)n3ccnc3)C2)csc1C 73745,CN1CC(O)CC1(C)C(=O)NCC1(CCNC(C2CNC(=O)C2)=O)CC1 73746,C#CC1(O)CCCN(C(C2CC2CNC(=O)C(CO)C(F)(F)F)=O)C1 73747,C1(OC)CC(F)CN(C(c2cnn(C3CCOCC3)c2)C(=O)NC(C)(C)C)C1 73748,CCCCC(CNC(=O)C(CC(F)F)N(C(=O)CN1CC2CC2C1)C)CCC 73749,N1(C(c2c(C)noc2C)=O)CC(C)(C)OC2(C1)CN(C(=O)CCc1nccs1)C2 73750,N1(C(C(CCC)N(C)C)=O)CCN(C(=O)C=Cc2cccc(F)c2Cl)C2CCC12 73751,CCC(C)C(C)N=c1[nH]c(=NCC2(c3cnccn3)CCC2)[nH]c2c1COCC2 73752,C=CCC(C(=O)NCC(CNC(c1cccc(C)c1[N+](=O)[O-])=O)OC)C(C)(C)C 73753,C(=O)(CS(=O)(=O)CCOC)N1CC(CC(=O)NC2C(OCC)CCC2)OCC1 73754,N1(C(C2C(C(C)=O)C2(C)C)=O)CCC(NC(=O)C(=O)NC2CC2)C(C)C1 73755,c1(C(=O)NCCSCC(=O)NC(C(C)(C)OC)C)c[nH]c(=S)cn1 73756,c1(CC)nc2ccccc2c(C(=O)NCc2c(F)cncc2Br)c1C 73757,C1(NC(CSCCCC)=O)C=CCN(C(=O)COC(C)=O)C1 73758,N1(C(C(CC(=C)C)NC(=O)Cc2ccon2)=O)CCN2C(=O)OCC2C1 73759,c1(CCCC(=O)NCC2CCN2Cc2ccccc2Br)ccccc1Cl 73760,c1(OCC)ccc(Cl)nc1C(=O)NC1CCN(c2ccccc2)C1 73761,C=C1CC2(C1)CC(C(=O)NC(C1CCCN(C(c3cc(N)cc(F)c3)=O)C1)C)C2 73762,C1(NC(Cc2ccc(C)cc2)=O)CCCC12CN(C(C1(C)CSC1)=O)C2 73763,c1(C(=O)NC(C2CCCC2)CNC(C2CC(OC)C2)=O)sc(SC)cc1C 73764,c1(C(=O)NC(C)CCNC(=O)CCC2CCCO2)ccccc1CO 73765,c1(CC(=O)NCC(C)(CO)NC(C(=Cc2cccnc2)C)=O)c(C)ncnc1O 73766,Cc1cnc(Cl)c(S(=O)(=O)Nc2ccc(C(=O)Nc3nccc(Br)c3O)nc2)c1 73767,c1(C(N2C(C(=O)NCc3nnc(C)n3C)CC3CC32)=O)cc(F)c(F)cc1F 73768,Cc1ccc(CC(N2CCC(C(C)C(=O)NCCCCN(C)C)C2)=O)cc1 73769,c1(C(=O)NCC2(C)CCN(C(=O)CC3COC(=O)N3)C2)ccc2nc(O)sc2c1 73770,c1(NC(c2nnnn2C)C)ccc(S(=O)(=O)NCCCC2CCOC2)c(Br)c1 73771,C1(C(N2CC(CCNC(C3CC4CC4C3)=O)(OC)C2)=O)CCN(C2CC2)CC1 73772,N1(C(C(C=C)(C)CC)=O)CCN(C(=O)C(O)C=CC)CC(C)(F)C1 73773,N1(C(c2c(OCC)scc2)=O)CCC(NCC(=C)Cl)C(C)C1 73774,Cc1[nH]cnc1C(=O)NCc1ncoc1C1CN(C(C2CC(CF)C2)=O)C1 73775,CCCCC(CNC(c1cncc(OC)n1)=O)NC(=O)C(CC)n1ccnc1 73776,C1(NC(C(C=CCCC)O)=O)CCN(C(c2ccncc2)=O)C12CCC2 73777,n1(CC)cc(CC(=O)N(C2(C(=O)NC3CCN(C(N)=O)C3)CC2)C2CC2)cn1 73778,CCCCCC(C)(C)C(=O)ON1CCOCC(O)(C(F)(F)F)C1 73779,Cc1cc(C#N)ccc1S(=O)(=O)N(C)C(C1(S(C)(=O)=O)CC1)C 73780,N1(C(C2(C#N)CC=CC2)=O)CC2CCN(C(C3CC3c3ccccc3)=O)C2C1 73781,C(=O)(CC(C)CC)N(C1(C(=O)NC(CCC)C2CC2)CCC1)C1CC1 73782,c1(C(N2C3C(C(N(C4(CCO)CC4)C)=O)C(C3)C2)=O)cc(O)nc(O)n1 73783,N1(C(c2oc(C)c(Br)c2)=O)CCC(C)C(NC(C2CCc3n[nH]cc3C2)=O)C1C 73784,C=CC(C)CCN=c1nc(-c2ccccc2)[nH]c(=NCc2ccc(Br)s2)[nH]1 73785,c1(C(=O)NC2C(NC(c3cc[nH]n3)=O)CCC2)ccnc2ccncc12 73786,N1(c2ccc(S(=O)(=O)NC(c3nccc(C)n3)C)s2)CCN2C(=O)CCC2C1 73787,C12(CSC)CC(C(=O)NCC(C(C)C)NC(=O)C=Cc3cncs3)(CO1)C2 73788,FC(F)=C1CCC(c2nnnn2CC(F)F)(NCC2CCC2CO)CC1 73789,c1(NCCNC(C)=O)ccc(S(=O)(=O)Nc2nc(Br)co2)cc1Cl 73790,CC(C)(CCC(=O)N1C2CCC1C(C(=O)NCCCc1cnccn1)C2)[N+](=O)[O-] 73791,CC(C)C(C#N)C(=O)NCCCC(=O)NCCC1CCC(C)O1 73792,C(=O)(C1Cc2ccc(F)cc21)NCC(CNC(C1(CCOC)CCCC1)=O)(C)O 73793,C1(O)(CNC(CCc2ccnc(C)n2)=O)CCN(C(=O)C2=CCCCO2)CC1 73794,C(CC(C)C)(C(=O)N1CC(C)CCC1CO)NC(C(C)NC(C)=O)=O 73795,C1(C(=O)NCC(CCOC)NC(=O)Cc2cnc[nH]2)COc2ccccc2C1 73796,c1(C(=O)NC2CCCC(N(C(=O)CCC#N)C)C2)ncc2cc(Cl)ccn12 73797,CON=CC(=O)NC(C)C(=O)NCC(=O)OC(C)C 73798,Cc1nnccc1C(=O)NC1CCC(CCNC(=O)CC2CNC(=O)O2)C1 73799,C(=O)(C(C)(C)C(C)C)NCCCC1OCCN(C(c2c(C)[nH][nH]c2=N)=O)C1 73800,N1(CC)CC2CC1CN(Cc1coc(-c3ccc(Cl)c(Cl)c3)n1)C2 73801,N1(C(C=C(COC)C)=O)CCC(NC(c2csc(-c3cnc[nH]3)n2)=O)C(F)C1 73802,N1(S(CCSC)(=O)=O)CC2CN(CCNC(=O)Cc3ccccc3I)CC2C1 73803,c1(C(=O)NC(c2n(C)ncc2)C(=O)NCCn2ccnc2)ncnc(O)c1F 73804,CCCCCCC(C)C(=O)NC1CC(C)(NC(=O)CCCN=[N+]=[N-])C1 73805,c1(C(=O)Nc2cccc(CNC(C(C)CC(N)=O)=O)c2)cnn2c(N)ccnc12 73806,C1(NC(=O)Cn2nccn2)CC2CC(NC(=O)CNC(=O)Cc3ccsc3)C1C2 73807,N1(C(C(COC)C)=O)CCC(NC(=O)Cc2csc(-c3ccco3)n2)C1C(C)C 73808,N1(CC(C)(C)NC(C(C=CCCC)O)=O)CCN(C(=O)CC(C)COC)CC1 73809,N1(C(c2c(OC)scc2)=O)CC2(CCN(C(=O)C(F)C(C)C)CC2)CC1C 73810,c1(C(N2CC(CC(C)NC(C(CC=C)C)=O)C2)=O)cnc(C(C)C)nc1C 73811,c1(CSC)noc(CCC(=O)NC2CC2CNC(=O)CC2CCCCO2)n1 73812,N1(C(c2snc(COC)n2)=O)CCC(c2n[nH]cc2F)CC1 73813,C(C(C(=O)N(CCS(C)(=O)=O)C)C(C)(C)C)NC(CC(C)C1CC1)=O 73814,CS(=O)(=O)c1ccc(C(O)CNC(=O)NCc2c(O)cccc2Cl)cc1 73815,CC12CCC(CNC(N3CCCOC(CCO)C3)=O)(CO1)C2 73816,c1(C(N2C(C)CC(CC(=O)N(C3CC4CC4C3)C)C2)=O)cnn2c1OCC2 73817,c1(CCNC(C(C)(C)OC(C)C)=O)ccc(CNC(C2CCC(=O)NC2)=O)cc1 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74151,CN1CCCN(C(=O)CC(C(F)F)NC(C2(C)CCN(C)C2)=O)CC1=O 74152,N1(C(c2c(C)cn(C)n2)=O)CCN(C(=O)Cc2ccc(Cl)nc2)CCC1C 74153,c1(N2CC3(CCN(C(CC(=O)N(C)C)=O)C3)C2)nc(Cl)nc2[nH]cnc12 74154,c1(NC(C2C(NC(C3CCC(=C)CC3)=O)C2)=O)ccc2ncsc2c1Br 74155,C(Cn1ccnn1)(C(=O)NOCCCOC)NC(C(CC)O)=O 74156,C1(NC(c2n(CCSC)nnn2)c2cnc(C(F)F)s2)CNC(=O)OC1 74157,C1(NC(CN(C(CN(C(C)=O)C)=O)CC2CC2)=O)CN(C)C2(CCC2)C1 74158,Cc1ccc(F)cc1CC(N1CC=CC(NC(c2occc2CN(C)C)=O)C1)=O 74159,Cc1ccc(C=CC(N2CC(F)CC2CNC(C2(C3CC3)CCCO2)=O)=O)o1 74160,C1(C(N(CCC)CCNC(C2(C(=O)OCC)CC2C)=O)=O)CNC(=O)N1C 74161,c1(-c2cn(C3(c4ccc(O)nc4)CCCC3)nn2)nc2ccc(Br)nc2[nH]1 74162,c1(CC)cc(C(=O)NCC2CN(C(=O)C(C)n3cccc3)CC2C)cn(C)c1=O 74163,n1(CC(=O)NC2(CN(C(c3ncn(CC)n3)=O)C)CC2)cnc2sccc2c1=O 74164,C1(NC(COCC#C)=O)CCN(C(=O)C(c2ccc(C)cc2)OC)CC1F 74165,CC(=O)C(C)CC(C)C(=O)NC1CC2(NC(=O)C(C3CCCCC3)O)COC1C2 74166,c1(NC(C)=O)ccc(C(=O)NCC2CCN2C(C2CCCCC2F)=O)cc1 74167,C1(C(N2CCC(C(=O)NC)C2C)=O)C2CCC(C2)N1C(c1cc[nH]c1C1CC1)=O 74168,c1(C(=O)NCCNC(CC(CCSC)O)=O)c[nH]c2ccc(Cl)cc2c1=O 74169,C1(C(C)CNC(=O)C(c2ccnn2C)O)CCN(C(C2(F)CCOC2)=O)CC1 74170,Cc1nc(C(C)C)[nH]c(=NC2CC(NC(=O)C(C(C)C)c3cccnc3)C2)c1Br 74171,C1(NC(C(=O)NCC(C(=O)OC)C)=O)CC2(CCCC2)C1 74172,c1(CC(CNC(CCC)CO)O)cccc(F)c1 74173,C1(CN(C(C(C)OCC=C)=O)CCOCCO)CCN(C(=O)CCCCC)CC1 74174,N(C)(C(=NCC(O)c1ccccc1Br)NCc1ccnn1C)CCCC 74175,N1(C(C=CSC)=O)C2CCC1CC(NC(c1ccc(C3(C)CC3(F)F)cc1)=O)C2 74176,c1(CC)nc(C(=O)N(C)CC2CCCN2C(=O)C=C(C)C(C)(C)C)cs1 74177,C1(C)(CNC(COCC#C)=O)CCC(NC(=O)COCc2nc[nH]n2)C1 74178,C1(C)(OCC(=O)NCCCN(C(c2cc(CC)no2)=O)C(C)C)CCOCC1 74179,N1(C(CC2N(CC)CCC2)=O)CCC(O)(CCNC(=O)C=CC(C)C)CC1 74180,c1(OC)cc(C(=O)Oc2nc3c(s2)CCC3)c(Cl)cn1 74181,Cn1ccc2c(CC(=O)NCC34CCC(CC3n3cc(CO)nn3)C4)cccc12 74182,NC(=O)CCC(=O)NC1CCCC(CNC(=O)Cc2coc(-c3cccs3)n2)C1 74183,N1(C(c2nc(C)n(C(F)F)c2)=O)CCC(C)(NC(=O)C(C)C(F)(F)F)CC1 74184,C1(=CC(=O)NCC(C(C)C)(C)NC(=O)C2=NOC(C)(C)C2)CCCCCC1(F)F 74185,c1(C(=O)NCC(C)NC(=O)CN2CCNC2=O)nnc(S)n1C 74186,CC(CC(C)(F)F)C(=O)N1CC(F)(F)CC1CCNC(=O)C(C)(C)c1cccs1 74187,C1(C(=O)Nc2cn(CCCC#N)nn2)(C(C)C)CCN(CC2C(CC(C)C)C2)C1 74188,C#Cc1cnncc1C(=O)NCC1(C)CCN(C(=O)C(C(C)C)SCC)CC1 74189,N1(C(C2C(CC)C2)=O)CCN(C(=O)C(n2ccnc2C)C)CC2(CC2)C1 74190,C1(NC(c2c(OC)cc(Cl)cc2)=O)CC(C)(C)C12CCC2 74191,C(=O)(C(O)CC(C)(C)C)N(C(C(=O)NCC=CCCC)C)C1CC1 74192,N#CC1CCC1C(=O)NC1CCCC1CNC(=O)C(O)C1CCC1 74193,S(=O)(=O)(CCCS(=O)(=O)N(C)C)N(C1CCCC1NC1CCC1(C)C)C 74194,CC(C(=O)NCC1CCN(C(=O)CSc2ccc(Cl)cc2)C1)C(C)(F)F 74195,CCCC(C)(CC)C(=O)N1CCC(CNC)C1.n12cc(nn1)C2 74196,c1(C(=O)NC(c2ccn(C)c2)=O)coc(C)c1.c1(C(CCCC)O)ccccc1 74197,c1(C(N2C(CCN(C(CC)=O)C)CCCC2)=O)cc(C)c(CO)cn1 74198,c1(CC)cccc(OCC(N2CC(O)(CN(C(=O)C=CC(C)CC)C)C2)=O)c1 74199,N1(C(C2C(CNC(=O)COc3cccnc3)OCC2)=O)CC2CCC2C1 74200,C(=O)(C1=CCCSC1)NCC(C)(O)CNC(=O)CNC(c1c(F)cccc1F)=O 74201,c1(CC(=O)NCC2(O)CN(C(C(CC)OCC)=O)C2)c[nH]c2cccc(Cl)c12 74202,N1(C(C(CC)(C)O)=O)CC2CCC2(CNC(=O)Cc2ccnnc2O)C1 74203,CC1CN(C(=O)COCc2ccccn2)CC(C)N1C(C1CC=CC1)=O 74204,C(C)(C)(CC(=O)NCC1(NC(=O)C(C2CCOCC2)F)CC1)OC 74205,C1(CC(=O)NC)CN(C(c2ccc(C)nc2)=O)CCN1C(=O)C#CC1CCC1 74206,c1(C(C(=O)NCCOC2CN(C(C(CCC)O)=O)C2)C)cccc(C#N)c1 74207,C(C(CC(=O)NCC1(C#N)CC1)C1CCC1)NC(c1c(C)[nH]cc1)=O 74208,C1(=O)CS(=O)(=O)N1C1COCC1O.c1(SC(C)(C)C)ccccc1O 74209,C1(C(=O)NC(C)CCNC(C2(C)CCC2)=O)C2CC1N(C(=O)OC(C)(C)C)C2 74210,c1(C(N2C(CNC(c3cn(CC)nc3)=O)CCC2)=O)cc(N)cc2c1OCCO2 74211,C1(C(=O)NCC(CNC(C2OCCN(C)C2=O)=O)O)(OC2CC2)CCC(C)(C)CC1 74212,N1(C(C2(N(C)C)CC2)=O)CC2CC(C1)C2NC(c1ccc(C(O)CF)cc1)=O 74213,C(N=c1[nH]cnc2c1COC2)C1N(C(=O)CC(F)(F)F)CCCC1 74214,c1(C(N2C(COC)(CNC(=O)C3=CCCC3)CCC2)=O)ccc2cccnc2c1 74215,C1(CNC(COc2c(C)cccc2)=O)N(C(=O)C(C)NC(N)=O)CCC1(C)C 74216,N1(C(CC(C)(C)C2CC2)=O)CC2CCC(C(=O)NCC3COC(=O)N3)(C2)C1 74217,C1(NC(C)=O)CCC(CC(=O)NCC(C2CCN(C(=O)C(C)(Cl)Cl)CC2)C)CC1 74218,C(=O)(C)NCCCNC(C)(C)C1(C(=O)OC)CC1 74219,C(=O)(C1=NNC(=O)CC1)N(CC(C)(C)NC(c1ccns1)=O)C 74220,C1(C(N2CC3(CCN(C(=O)CC4CCCO4)C3)C2)=O)CCCCC(F)(F)C1 74221,N1(C(C2(CNC(=O)CC3(O)CCCC3)CC2)=O)CC2CC2C2CC12 74222,C(=O)(C(CC)C(=O)NCC1CN(C(=O)C(C)(C)O)CC12CC2)OCC 74223,C1(NC(C2CSCCS2)=O)CN(C(C2CC(O)C2)=O)CC1n1cccn1 74224,c1(C(=O)NC2C(C)CN(C(=O)C#CC3CC3)C2)ccc2ccoc2c1 74225,CCCCC(C(=O)NCC(C(C)(C)C)OC)NC(c1cc(C)c(C)[nH]1)=O 74226,c1(NCCC2C(CC)C2)cc(N2CCC(COC)C2c2ccccc2)ncn1 74227,Cc1nc(C(N2CC(CNC(=O)C(=Cc3c[nH]cn3)F)C2)=O)nn1C 74228,C1(C(N2CC(CC(C)C)OCC2)=O)CC(C)(C)CCN1C(=O)C1=C(Cl)CCC1 74229,N1(C(CSCCCC)=O)CC(NC(c2cc(O)nc(C3CC3)n2)=O)CC(F)C1 74230,N1(C(C(C)(C)C#N)=O)CC2(CCC(CNC(C3CCC4CC34)=O)O2)C1 74231,C(CC(C)(O)C(=O)NC1CCCC(N2CCCC2=O)C1)C1(C)CC1 74232,CC1CCCn2c(CC(=O)NC3CCCCC3Oc3ccccc3F)cnc21 74233,C(CCC(C)C)(C(=O)NCCC(C)(C)C)NC(c1c(C)cccn1)=O 74234,c1(-c2c(C(=O)NCC(CC)NC(=O)CCC(C)=O)c[nH]n2)cc(F)cc(F)c1 74235,Cc1nc(NCc2cccnc2-n2cccn2)cc(N2CCC(CO)C2)n1 74236,n1(C(CC)CC)nc(-c2cccc(N)n2)nc1C1CC1OC(C)(C)C 74237,c1(C(=O)NCC(CC)NC(C2CCC(=O)N(C)C2)=O)[nH]c2cc(C)ccc2c1C 74238,N1(C(C(C)N(C)C)=O)CCC(NCc2cnn(C)c2)C1 74239,c1(NC(=O)NC(c2ccc(OC)cn2)C)nc2c(s1)CCc1ccccc1-2 74240,C1(C(=O)NC(C2CCCCC2)C(C)NC(C(OC)OC)=O)CN(C)CCN(C)C1 74241,C1(C(=O)NCc2c(C(=O)NC(CC=C)CC=C)scc2)CC2(C1)CC2(F)F 74242,c1(C(=O)NCCC2(O)CN(C(c3ccon3)=O)C2)cc(Br)ccc1Cl 74243,c1(C(=O)NC2C(NC(CC(CC)C3CC3)=O)CCC2)cn2nc(OC)ccc2n1 74244,CCCCC(CC(=O)NCC1(COC)CCCC1)NC(=O)CNC(=O)C(C)(C)C 74245,S(=O)(=O)(c1ncn(-c2ccccc2)n1)N(CC)Cc1ccoc1 74246,C1(CC(=O)N(CC(=O)NCCOC)C)SC(=Nc2ccccc2)NC1=O 74247,CCC(C)(C(=O)N1CCC(NC(=O)COC2CC(F)(F)C2)CC1)OC 74248,N1(C(CCCOCC=C)=O)CCCC(O)(CCNC(=O)CC(O)C(C)C)C1 74249,C(=O)(C(O)C(C)SC)NC1(CC=C)CN(C(=O)C(=O)Nc2ccc(Cl)cc2)C1 74250,N1(C(CC2(C)CCN(C(c3noc(CC)c3C)=O)C2)=O)CC2(C1)CC2(F)F 74251,C1(C)(CNC(CNC(C)=O)=O)CN(Cc2ccc(Cl)cc2Cl)CCO1 74252,Cc1ccc(F)c(CC(=O)NC2CCN(C(=O)C(C)CC(N)=O)CC2O)c1 74253,N1(C(CC2ON=C(CC)C2)=O)CCC2CN(C(c3cncnc3CC)=O)CC2C1 74254,C(C(CC)(CC)CO)NC(C1N(C(C(CC)COC)=O)CCCC1)=O 74255,CN1CCN(C(=O)CSCc2ncc[nH]2)C(CNC(=O)Cc2cncnc2)C1 74256,c1(C(CC(=O)N(CCC(CC)O)Cc2ccccc2)NC)ccc(F)nc1 74257,N1(C(CNC(C=C)=O)=O)CCN(C(c2cc(-c3ccc(C)cc3)no2)=O)CC1C 74258,O(P(=O)(OCC)C(F)C(=O)NCC1CCc2nn(C)cc2C1)CC 74259,c1(C(=O)OC)cc(NC2CC(C(F)F)C2)cc(Cl)c1 74260,N1(C(Cn2c(C)nnn2)=O)CCCC12CCC(NC(=O)C(CO)N(C)C)CC2 74261,CN1CC2CCN(C(=O)C(CCC3CC3)NC(=O)CCC3CC3(F)F)CC2C1 74262,Cc1cn(C)cc1C(=O)NC1CC(CNC(=O)CC2(C)CCCO2)C1 74263,c1(OC)cc(OC)cc(C(=O)NCCN(C2CCCC2)C(=O)CC2CC2C)c1 74264,c1(OCC#C)ncccc1C(N1CCC(OCCc2c(C(=O)NCC)csn2)C1)=O 74265,N1(CCCc2ccc(C)cc2C)CCc2ccc(C(=O)O)cc2C1 74266,c1(C(N(C(C)CNC(=O)C(C(C)C)n2ccnc2)CC)=O)snc(O)c1Cl 74267,c1(C(CNC(=O)COC(F)F)NC(c2ccoc2C2CC2)=O)cccc(Cl)c1 74268,c1(CC)nc(O)c(C(N2CCC(NC(=O)C(C)OCCN(C)C)C2)=O)cc1C 74269,C1(n2cc(CNC(C)=O)nn2)CN(C(c2ccc(C(C)C)cn2)=O)CC1C 74270,N1(C(CCN(C(C2CC(OCC)C2)=O)C(C)C)=O)CCOCC1C1(C)CC1 74271,C=C(C)C(C)(C)C(=O)N1CCC(Cn2cc(CNC(=O)N(C)C)nn2)C1 74272,Brc1cc(I)ccc1CNC1(c2nnnn2Cc2ccccc2)CCC2CCC12 74273,C(=O)(CC1C(=O)Nc2ccccc21)NCC1CN(C(C2CC(=C)C2)=O)C(C)C1 74274,Cc1ccc(=N)[nH]c1C(=O)N(C(C)CNC(c1ccn(C2CC2(F)F)n1)=O)C 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74556,C12(CNC(c3cnsc3)=O)CN(C(C3CC4(CC4)CO3)=O)CC1CCO2 74557,c1(CC)nc(C)ccc1NC(C1COCCC1NC(=O)CCN=[N+]=[N-])=O 74558,C12(C(N3CC(CC)OCC3)=O)COCC1CN(C(=O)Cc1[nH]cnc1C)C2 74559,c1(C(N2CC(O)(CNC(C(C(CC)O)C)=O)C2)=O)cc2sccc2n1C 74560,c1(C(N2C3CC(NC(C(C4CC4)OCC)=O)C2CC3)=O)c(F)cccc1[N+](=O)[O-] 74561,C1(CC(=O)NC(CC)CNC(C2CCCCS2)=O)CCC2(CC1)CC2 74562,C1(CN(C)C(C2CCCN(C(N)=O)C2)=O)CCN(c2ncncc2Cl)CC1 74563,c1(N2CC(C)C(CS(N)(=O)=O)C2)nccc(=NCc2cncn2C2CC2)[nH]1 74564,C=CCCCCCC(=O)N(C1CC(NC(=O)CCNC(=O)NC)C1)C 74565,Cc1ncnc(C)c1C(N1CCN(C(=O)CC(=O)NCC(F)(F)F)C(C)C1)=O 74566,c1(C(=O)NCC(CN(C(=O)C(O)c2ccsc2)C)O)cc(N)c(F)c(O)c1F 74567,Cc1cc(CC(=O)NC2(CNC(c3nocc3C)=O)CCC2)cc(F)c1 74568,C1(C(=O)OCC)(CC)CCN(CC(=O)NC(C)CNC(C2CCOC2)=O)CC1 74569,c1(C(C(=O)NC(CNC(CN(C)CCO)=O)(C)C)(F)F)cc(Br)ccn1 74570,N1(C(C=CCN(C(=O)C(c2ccccc2)F)C)=O)CC2CCC(C1)C(=O)O2 74571,c1(OC)ccc(O)cc1CNC(=O)CCn1cc(CN(C)CCO)nn1 74572,C1(O)(CNCC(COc2ccc(CCOCC)cc2)O)CCCCCC1 74573,C1(C(=O)NC2CC(=O)NCC2)CCCCCC1NC(C1(CO)CCCO1)=O 74574,N1(C(c2c(C)scn2)=O)CCCC(C2CCCCN2C(c2sccc2Cl)=O)C1 74575,N1(C(C2(OC)CC2)=O)CC2CCN(C(c3cc(C(C)=O)c(C)o3)=O)C2C1 74576,CCCC(C(O)C(=O)NOC1CCCN(CC)C1)NC(=O)CNC(=O)C(C)CC 74577,C(=O)(CC(c1ccccc1)N(C(c1ccc[nH]1)=O)C1CC1)NC(c1cccs1)C 74578,C1(CC#C)(C(=O)N(C2CCN(C(=O)C=CC3CC3)C2)C)CCCCO1 74579,N1(C(c2cccc(CCC)c2)=O)CCC2(N(C(C3CCC3)=O)CC)CC2C1 74580,c1(C(=O)NC(CNC(c2n(CCC)ncc2)=O)CO)ccc(C(C)C)nc1 74581,C1(CNC(c2c(CC)n[nH]c2)=O)CN(C(=O)C(c2c(C)noc2C)C)CCCO1 74582,c1(C(=O)NCC2(O)CCN(C(CC(CC)OC)=O)C2)cccc2nsnc12 74583,Cc1noc(C(=O)O)c1Br.c12sccc1NC(=O)CC1(C)CN(C1)C2 74584,CN1CC(C(=O)NCC2(NC(=O)C(CN(C)C)N(C)C)CCCCC2)CC1=O 74585,C(=O)(C(CCC1CC1)NC(=O)CC(N)=O)NC1C(c2n(C)ncc2)C1 74586,C1(NC(CC2CCCN(C(C(C)c3cc[nH]n3)=O)C2)=O)CCC(=O)NC1(C)C 74587,N1(C(C2N(C)CCC2)=O)CCC(O)C2(CCN(C(c3c(I)cnn3C)=O)CC2)C1 74588,CC1=C(C(=O)NC2CC(F)CN(C(=O)Cc3cnoc3)C2)Cn2ncnc2N1C 74589,C12(NC(c3c(C)nc(CO)s3)=O)CCCC1N(C(=O)C(C1CCCCC1)F)CC2 74590,C1(CNC(Cc2cncc(C)c2)=O)CCCCN(C(c2cccnc2O)=O)C1 74591,c1(C(=O)NC2(CCC(N3CCN(C(=O)OC)CC3)=O)CCC2)c[nH]c(C#N)c1C 74592,Cc1ccnc(C(=O)NC2CCC(C)(CNC(c3sccc3CC#N)=O)C2)c1 74593,c1(OCC)cc(Cl)c(Br)cc1C(C(=O)NCCCF)N(CCC#N)C1CC1 74594,C1(CC(=O)NCCN2CCN(C(C3CCC(O)CC3)=O)CC2)CC2CCC(C1)C2 74595,CC1(C)CN(C(C2CC(F)(F)CN2C(c2ccc([N+](=O)[O-])o2)=O)=O)CCO1 74596,C12(CCNC(c3cnc(OC)s3)=O)CCC1CN(C(C1(F)CCN(C)CC1)=O)C2 74597,N1(C(C2CCN(C(CNC(=O)OCC)=O)C2)=O)CCSCC1C 74598,C(=O)(C(C)(C)C(F)(F)F)NCC1C(CC)CN(C(=O)C(C)C2CCCO2)CC1 74599,C1(NC(N2CCC(c3nccn3C)(OC)C2)=O)Cc2ccccc2OC1C 74600,C1(O)(CNC(Cc2cnc(C)[nH]2)=O)CCCN(C(C2CNC(=O)N2C)=O)CC1 74601,c1(-c2cn(CCCCCC)nn2)ccccc1C(=O)NC 74602,N1(Cc2ccc(C(=O)OCC)cc2)CCC2(CC1)CS(=O)(=O)CCO2 74603,c1(C(=O)NCC(CC=C)NC(C2CC2C(C)C)=O)cc(N)cc(O)c1 74604,c1(C(=O)C(C)=O)cc(OC)n(C)n1.C12CCCN1C2=O.C12CC(C1)NC2=O.CO 74605,N1(C(C2C(C)CCOC2)=O)CCN(C(c2ccn(C(C)(C)C)c2)=O)CC1CO 74606,c1(-c2n(C(CC)C)nc(COc3ccc(OC)cc3)n2)nccn2nc(C)cc12 74607,CCCCC(CC(=O)NCC1(CO)CC2CC2C1)NC(c1ccc(C)nc1O)=O 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74625,C1(NC(CCCC=C)=O)CC2(CCN(C(C3(C(C)C)CC3)=O)C2)C1 74626,c1(C(=O)NC2C(OC)CN(C(CCCOCCC)=O)C2)cnn2ccn(C)c12 74627,CCCCCC(O)C(=O)N1CCC(C)CC1C(N1CCC1C(=O)NCC1CC1)=O 74628,N1(C(CC(=O)NCC#C)=O)CCOCCC1C(=O)NCC1CC(C(N)=O)=NO1 74629,C1(O)(C(c2n(C(C)(C)C)nnn2)NC2CN(c3ccccc3)C2)CCCCCC1 74630,N1(C(c2c(C)snn2)=O)CC2CCC1C(NC(c1n[nH]cc1[N+](=O)[O-])=O)C2 74631,C(CC(C(=O)NC1(C(=O)NCC(O)COC)CCCC1)OC)OC 74632,N1(C(C(COC)N(C)C)=O)CCOCCC1C(=O)NCC1CC2(CCCO2)C1 74633,CC1(C(N2CCC(C)(CNC(C3CC(F)(CF)C3)=O)CC2)=O)CCC2CC2C1 74634,C(C(N=[N+]=[N-])C(=O)NCCCC(C)NC(c1csc(CC(C)C)n1)=O)OCC 74635,C1(NC(C(C(C)C)OC)=O)CC2CCC1CN(C(C1(O)CCCCCC1)=O)C2 74636,C(=O)(C(C)(C)C1CCCN1C(=O)CCN(C)C)NC1(C(C)C)CC1 74637,Cc1nsc(N)c1-c1cn(CC(=O)NC(C2(O)CCC2)C2CC2)nn1 74638,C1(CNC(c2n(C)ccc2)=O)CC2(CN1C(=O)C=CC1CCCCC1)CC2(F)F 74639,C1(NC(c2c(CC)nco2)=O)CCCCC1CNC(=O)C(O)CC1CCCC1 74640,C1(C2CCN(C(C3CCN(c4nccs4)CC3)=O)C2)(NC(C2CCSC2)=O)CC1 74641,Cc1cc(C(N2CCCCC(NC(c3ncncc3C)=O)C2)=O)c(Cl)cn1 74642,CC(C)C(C(=O)NC1COCCC1NC(C1CC(O)(C(F)(F)F)C1)=O)C(C)C 74643,C(C(O)CC(=O)N1CC(N(C)CCO)C1)NC(CSCC=C)=O 74644,C(=O)(C1=CC2CCCC12)N(C1CCN(C(C2(SCC)CC2)=O)CC1)CC1CC1 74645,Cc1noc(Cl)c1CC(=O)NC1CCC(CNC(C2(C)CCOCC2)=O)C1 74646,c1(OC)cc(-c2nnc(C(=O)OC3CCCCO3)s2)cc(OC)c1OC 74647,N12CCCCC1CNC(=O)C2=O.n1(CC)nnc(Br)c1C(F)F 74648,C=C(Cl)C(C)(C)C(=O)NC(CNC(=O)C(c1ccc(Cl)cc1)(C)O)C1CC1 74649,n1(CCCC(=O)NCC2CCN2C(C2CCCCCC2)=O)ccccc1=O 74650,CC#CCCC(=O)NCCC1CC(CNC(=O)C(CCSC)NC(=O)CCC)C1 74651,N1(C(c2c(C)cc(C)o2)=O)CCC(NC(=O)C=C=C(Cl)Cl)C(C)(C)C1 74652,N1(C(c2cc(OC)cc(OC)n2)=O)CCC2CN(C(=O)Cc3ccsc3)CC12 74653,CC(=O)CCCC(=O)N1CCCC(NC(=O)C(C)CC2CCCC2)C1 74654,c1(N2CC(c3ccccc3)=C(C)C2)nc(C)c2ncn(-c3cccc(C)n3)c2n1 74655,C(=O)(C#CC1CCOC1)NC(CCCC)CNC(=O)CC1(NC(C)=O)CC1 74656,C1(NC(=O)NC(c2ccc(Br)s2)C)CCS(=O)C1 74657,C(=O)(C1=CS(=O)CCC1)N(C1CCCN(C(CCn2ncc(C)c2)=O)C1)CCO 74658,CC1CCN(C(c2c[nH]c(=N)o2)=O)CC1NC(=O)CC1CC(=O)NC1=O 74659,n1(CC(=O)NC2(CO)CCN(C(=O)C(c3ccc(F)cc3)F)C2)ccccc1=O 74660,C(=O)(CCCCCF)NCC1C(NC(=O)CSCc2ccccc2Cl)C1 74661,Cc1cc(C(=O)NCC2C3CC2N(C(c2conc2C2CC2)=O)C3)cc(=O)n1C 74662,CCC1CNC1=O.c1(-c2cn(CCCOC)nn2)cc[nH]c1C(=O)O 74663,c1(C(=O)NC(C2CCCO2)CC)cncc(CNC(=O)C(C)c2ccco2)c1 74664,C1(NC(C2(CC#C)CCCC2)=O)CCCN(C(=O)Cc2ccc(Cl)cc2C)C1C 74665,Cc1cc(C)c([N+](=O)[O-])c(C)c1CN1CCN(CCC2COC2)CC1 74666,N1(C(c2nc(CCC)sc2)=O)CCC(CN(C(=O)CC(=O)OC(C)(C)C)C)CC1 74667,N1(C(c2ccc(=NC)[nH]c2)=O)CCCC2CCCC(O)C12 74668,C(CC(C)C)(C(=O)N(C(C)CN(C)C(c1ccncc1C)=O)C)OC 74669,CC(C)(C)CS(=O)(=O)NCCC1(O)CC2CCC1C2 74670,C1(CCOC)(NC(c2cn(CCCC)nn2)=O)CCN(C(C2CC(=O)CO2)=O)C1 74671,N1(C(CCC)=O)CCn2ncc(CN(C)C(c3cccc(Cl)c3F)=O)c2C1 74672,Cc1cccc2c1CCN2C(=O)CCOCCNC(=O)CC(C)CC(C)C 74673,c1(C(=O)NC(C2(O)CN(C(C=CCC)=O)C2)C)cccc(OC2CCCC2)c1 74674,c1(C(=O)NC2C=CCN(C(=O)CC34COC(CF)(C3)C4)C2)cnc(F)c(F)c1 74675,C(c1ccccc1Br)=CC(=O)NCC1(C)CCC(NC(c2ccc[nH]2)=O)C1 74676,Cc1ccc(C=CC(=O)NCC2(NC(C3CCN(C)C3)=O)CCC2)nc1 74677,N1(C(C=CCC)=O)CC(C)(C)C(NC(c2cc(CO)[nH]n2)=O)C(C)(C)C1 74678,c1(C(N2C(CN(C(=O)C(C)O)CC)CCCC2)=O)ccc(C)c(F)c1N 74679,Cc1cc(C(N2CCC(C)(NC(c3cc(O)nc(O)c3)=O)C2)=O)c(Cl)cc1F 74680,CCCCC(O)C(C)C(=O)NC(C(=O)NC1CC(C)N(C)CC1C)C1CCC1 74681,N1(C(CC2(COC)CC2)=O)CCC(C(=O)N(C2CCC2(C)C)C)CC1 74682,c1(OC)cc(C(C)NC2CCCN(c3ccncn3)C2)ccc1OCCO 74683,N1(C(CC(CN(C)C)O)=O)CCC(C)(C)C(CNC(c2[nH]nnc2C2CC2)=O)C1 74684,c1(OCC)ccc(C=CC(N2CC(CNC(C3(F)CC3)=O)CC2C)=O)cc1OC 74685,c1(C(=O)NC2CN(C(c3c(C)ncs3)=O)C2)cccc(Cl)c1F 74686,C1(CC(C)NC(C2CCC(=O)O2)=O)CCN(C(C2C3COCC23)=O)CC1 74687,C(=O)(C(C)C(C)CC)N(CC(=O)NC1(CO)CCC(C)C1)CC#C 74688,N1(C(C=CCCC)=O)CCN(C(C2CC(=C(F)F)C2)=O)CC1c1ccccc1 74689,C1(CC#C)CCN(C(c2ncoc2CNC(C2CC2CCC)=O)=O)CC1 74690,c1(C(N2CCC(N(C(CC(CC)SC)=O)CCO)C2)=O)ccc(C)nc1C(C)C 74691,N1(C(c2c(C)nc(O)cc2)=O)CC2CCC1CC2NC(c1cnc[nH]1)=O 74692,S(=O)(=O)(c1ccc(Cl)c(Cl)c1)NCCNC(CCCC(N)=O)=O 74693,C1(NC(C(C)(C)OC)=O)CCCN(C(c2sc(-c3ccsc3)nc2C)=O)CC1F 74694,C(c1ccc(O)c(OC)c1)=CC(=O)N(CCCN(C(C(C)SC)=O)C)C 74695,N1(C(c2c(C)cc(C)o2)=O)CCC2CN(C(=O)CC3(O)CCCCCC3)CC12 74696,N1(C(C(C)C)=O)CCN(Cc2cc(Cl)ccc2Br)CC1C(F)(F)F 74697,N1(C(C2(c3cc(C)no3)CC2)=O)CC2CC(NC(=O)C(C)C3CC3)CC2C1.OC=O.C 74698,Cn1c(C(=O)NC2CCC(CCNC(c3c[nH]c(=N)s3)=O)C2)cc(Cl)c1Cl 74699,N1(C(C2CC(C)OCC2)=O)CCCC2(C1)CN(C(=O)Cc1cncn1C)CCO2 74700,c1(NC(c2c(CNC(C=C(C)C(F)F)=O)n[nH]c2)=O)ccc(OCF)cc1O 74701,CN1CCCCC(C(N2CCOC(CNC(C34CCC(C3)C4)=O)CC2)=O)C1=O 74702,C(=O)(CCN(OC)C(=O)c1cnnc(C)c1C)NCC(CC)(C)C 74703,c1(CC)cnc(O)c(C(N2CC(NC(=O)CCc3ncco3)CC(C)C2)=O)c1 74704,C1(CNC(c2cc(C(C)C)[nH]n2)=O)CC(C)CCN1C(=O)CCn1cc(Cl)cn1 74705,O=S(=O)(c1cc(F)cc(F)c1)NCC1CCCCN1Cc1nc2ccccc2[nH]1 74706,c1(C(=O)NC(CCNC(C(CC=CCC)C)=O)(C)C)ccc(=O)n(CCOC)c1 74707,c1(-n2cc(CN3Cc4c(nc(C)s4)C3)nn2)ccc2c(c1)NCCC2 74708,Cc1ccc(C(N2CC=CC2C(=O)NC(C)CCC(C)C)=O)c(O)c1 74709,N1(CC)CCN(C(=O)C(C(C)C)NC(=O)C(CSC)OC)CC1 74710,C1(NC(C2OCCN(CC)C2)=O)CN(C(=O)CSCCOC)CCC12CCC2 74711,C=C(Cl)C(C)(C)C(=O)NC(CNC(=O)C(c1ccc(C)cc1)C1CC1)CC(C)C 74712,C12(CNC(CC(C=C)C)=O)CC(CC)(CN1C(=O)C(CCOC)OC)C2 74713,c1(C(=O)NCC(C2CCCC2)NC(c2ccoc2Cl)=O)ccc2oc(O)nc2c1 74714,C1(SCCC(=O)N(CC(C)N(C(=O)COCC(C)(C)C)C)C)CCOCC1 74715,c1(N(C(=O)C(C)(C)C)C)nc(C(N2CCCC2c2nn[nH]n2)=O)cs1.C1C(=O)N1 74716,CC1CC(NC(c2cncn2-c2ccccc2)=O)CN1C(=O)C=CC1CCCC1 74717,N1(C(C)=O)CS(=O)(=O)CC1C(=O)NCC(C)(C)CN(C(=O)CCCCC1CC1)C 74718,C(=O)(C1OCCn2ccnc21)NC(C)CCCNC(c1csnn1)=O 74719,c1(C(=O)NCCCOCCCNC(C(CC)(C)C)=O)cn2c(n1)C(C)CCC2 74720,C1(C2CN(C(c3ccc(C(F)F)s3)=O)C2)(NC(=O)COC2CCCCCC2)CC1 74721,C(=O)CCCC(F)(F)CO.N1(c2n(C)ncc2)CCCC(c2nn[nH]n2)C1 74722,c1(C(=O)NCCOCCNC(C2CC(O)(C(F)(F)F)C2)=O)c(CO)cccc1F 74723,C1(O)(CNC(=O)Cc2csc(S)n2)CCCN(C(C2CCC=CO2)=O)C1 74724,N(C1CCCn2nccc21)C(CC1N(C(CCC(CC)C)=O)CC2(CC2)C1)=O 74725,Cc1ccnc(O)c1C(N1CC2C(C(=O)NC(C)CN(C)C)C2C1)=O 74726,c1(NCC2(F)CC(C(=O)NC(Cc3cn(C)nc3)=O)C2)cc2cc(F)ccc2s1 74727,c1(C(=O)NCC23N(c4nccc(OCC)n4)CC(C2)C3)nc(O)nc(O)c1OC 74728,N(C1CCc2c(Br)ccc(Cl)c21)CC1CC(O)C1 74729,c1(OC)ccc2cc(C(=O)NC(C3CN(C(c4oncc4C)=O)C3)C)ncc2c1 74730,c1(CNC(CC(COC)NC(c2n[nH]cc2C)=O)=O)c(C)cccc1C 74731,CC(N=c1[nH]c2c(c(=NC3CC(C4CC(F)(F)C4)C3)[nH]1)COCC2)c1ccsc1 74732,c1(C(=O)NC(CN(C(c2ccc(SC)o2)=O)CC)C)cn2c(n1)CC(OC)CC2 74733,c1(C(C)NC(=O)NC2CCOC2c2ccccc2)cccc2cccnc12 74734,C1(CNC(C2C(C)(C)OCC2)=O)COCCN(C(C23CC(C2)C3)=O)C1 74735,C(=O)(C1=CC(C)(C)C1)N1CCC(NC(c2cn(CCC)nc2)=O)(COC)C1 74736,c1(NCC2(CSC)CCC2)ccc(S(=O)(=O)N(C)CCO)c(Br)c1 74737,C1(C(=O)NCc2ccc(OCC=C)cc2)(NC)CCOC(C)(C)C1 74738,CC1Cn2nccc2CN1C(=O)C1=CCCN(C(=O)COCCCF)C1 74739,N1(C(C(C)OCC=C)=O)CC(O)CC1CNC(=O)C1=COCC1 74740,c1(CC(N2C(CNC(C3C(C(C)C)C3)=O)CC2)=O)cnc2ccccc2c1 74741,C1(N(C)C(c2ccc(Cl)s2)=O)CCCN(C(=O)CC23COC(CF)(C2)C3)CC1 74742,Cc1cc(NC(C2CCN(C(=O)OC(C)(C)C)C2C)=O)c(C)n1Cc1ccccc1 74743,C(=O)(C(C)C(O)C(C)C)N1CCC(NC(CC(C)=C(C)C)=O)C(O)C1 74744,c1(CC)cccc2[nH]c(C(N3CC4CCCC3(COc3ccccc3)C4)=O)cc12 74745,C1(F)(C(c2ccccc2)=O)CN(CC(C2CCCOC2)=O)CC12COC2 74746,c1(C(=O)NCC2CCCN(C(C(C(C)C)C)=O)C2)c(F)ccc(Br)c1F 74747,CC1CCN(C(=O)C(O)C2CCCC2)C1CNC(C1CCCSS1)=O 74748,CC1C(NC(=O)CC2(C)CCCO2)CCN1C(c1cccc(Cl)n1)=O 74749,CC(Cc1cnc[nH]1)C(=O)NCCN(C(C1CCOC1c1cn[nH]c1)=O)C1CC1 74750,C1(NC(c2c(CC)cns2)=O)CC(O)CN(C(c2cnccc2Cl)=O)C1 74751,c1(N(C)Cc2ccc(-c3c(OCC)cccn3)s2)ccc(S(=N)(=O)CC)cc1 74752,C(C1=NOC2CN(C(=O)CCC3CCCCC3)CC12)NC(C12OCC(C)(C1)C2)=O 74753,C1(C2CC2)C(CC)CCCN1OC(CC1CCN(C(C2C(C)C2C)=O)C1)=O 74754,C1(CC)CC(C(N2CCC(CCNC(=O)CC(C)F)CC2)=O)CC(=O)N1 74755,CC(C)CC(CNC(C1(NC(=O)C(c2ccnn2C)C)CCOCC1)=O)CO 74756,c1(NC2C(NC(c3cccc(Br)n3)=O)CCC2)ncnc2occc12 74757,N1(C(c2c(Cl)ccc(NC)c2)=O)CCC2CCCC(C1)N2C(=O)C(C)SC 74758,C1(C(=O)NCCCN(C2CC2)Cc2c(CC)noc2C)CCc2nncn2CC1 74759,c1(C(N(C2CCN(c3ccncn3)C2)CC)=O)ccc(=O)n(C2CC2)c1 74760,N1(C(C2C(CNC(c3cccc4c[nH]nc34)=O)C2)=O)CCN2C(=O)NCC2C1 74761,N1(CC(=O)NC(C)(Cn2cccn2)CO)CCCN(CC(=O)NCN)CC1 74762,n1(CCOC)c(N(CC(=O)Nc2cc(Br)cs2)C)nnc1C1CCCc2ccccc21 74763,C1(CNC(c2c(C(C)C)nco2)=O)CCCCN(C(=O)CCC2CC(F)(F)C2)C1 74764,C(N=c1nc(C)c(Br)c[nH]1)C1(O)CN(C(CSc2nc(C)cc(C)n2)=O)C1 74765,C1(CNC(C2CN(C(N)=O)C2)=O)C=CCN(C(=O)CCc2nc(C3CC3)no2)C1 74766,C1(OCC)CC2(C1)CC2C(=O)NCCC1CCN(c2nnc(C(F)F)o2)CC1 74767,C1(Cc2n(-c3n(C)ccn3)nc(C(F)F)n2)CCc2ncsc2C1 74768,C1(CNC(C2(COC)CCC2)=O)CCCCCN1C(c1ccc(O)nn1)=O 74769,N1(C(c2ccc(SC)s2)=O)Cc2ccc(-c3ccc(O)cc3C)cc2C1 74770,C1(CCOC)(NC(COCCC=C)=O)CCN(C(c2snnc2CC)=O)C1 74771,C1(CNC(Cc2cccc(C)c2)=O)C(C2CC2)CCN1C(=O)Cn1cncn1 74772,C(=O)(C(CC)CC(F)F)N1CCN(C(C2C(CC)CCC2)=O)CC1C1CCC1 74773,C(=O)(CCCN=c1nccc[nH]1)NCCC(C)NC(c1ccn2ccnc2n1)=O 74774,N1(S(c2ccc(C(N(C)C)=O)cc2)(=O)=O)CC2(CCOCC2)CC1CO 74775,c1(CCC)ccccc1C(=O)NC1CN(Cc2ccc(C(C)C)cc2)CC1O 74776,Cc1cc(C(=O)NCc2ncoc2CCNC(C2CCC(=O)C2)=O)c(Cl)cc1F 74777,CC1Oc2ccccc2OC1C(=O)NC1COCCN(C(=O)CN(C)C)C1 74778,CC(C)CC(F)C(=O)N1CCN(C(c2snc(Cl)c2Cl)=O)CC1CCO 74779,c1(C(N2CC=CC(NC(C=C(C)Cl)=O)C2)=O)cc(F)cc2nccnc12 74780,C1(C(=O)NC2CN(C(C(CC(C)C)=O)=O)C(C)CC2)CCOC2(CCC2)C1 74781,C(CCC(=O)NC(C)(CNC(=O)CNS(=O)(=O)CC)CC)=CC 74782,c1(C(=O)NCC2CCC(C)CN2C(C23CCN(CC2)C3)=O)cccc2[nH]ncc12 74783,C1(CC)(NC(=O)C(CCC2CC2)NC(=O)COCCCF)CCNC1=O 74784,C1(NC(c2c(C)c(N)ccc2)=O)CC2CC1CN(C(C1CCC(C(N)=O)C1)=O)C2 74785,c1(CN2C(C)(C(=O)Nc3cc(OC)c(Br)nc3)CC2)ccc(F)c2ccccc12 74786,CC1(C(=O)NCc2ccccc2)CCN(C(c2ccncc2)=O)C1 74787,C1(C(N2CC(CNC(c3ccc(C(=O)CF)cc3)=O)C2)=O)CC2(C1)CC(F)C2 74788,Cc1ccc(C(N2CC3C(NC(=O)Cn4cnnc4O)C3C2)=O)cc1S(C)(=O)=O 74789,C(CCCC(C)NC(=O)CC1(C(F)F)CC1)NC(c1c(C(=O)OCC)con1)=O 74790,c1(OC)c(C(N2CC(NC(c3cc(C)c(C)[nH]3)=O)C(C)(C)C2)=O)cc(Cl)cc1Cl 74791,C1(C(C)C)OCCC1CNC(=O)C(CO)NC(=O)CC(C)n1cccn1 74792,C(=O)(CCN(OC)C(=O)C1CN(C)CCO1)NC(CC)C(N)=O 74793,c1(OC)ccc(CC(=O)NCCC(C)NC(c2cnc(C(C)(C)C)s2)=O)cc1 74794,C(=O)(CC(CC)CC)OC(CCC)CN1C2CCC1COC2 74795,C1(NC(C2N(C(C)=O)CCC2)=O)C=CCN(C(=O)CSc2cnn(C)c2)C1 74796,C1(NC(CC(COC)C)=O)CN(C(c2conc2C(C)C)=O)Cc2ccnn2C1 74797,C1(NC(CC=C)=O)C2CCN(C(=O)C(c3ccc(F)cc3)(F)F)CCC12 74798,C1(CC(=O)N(CCNC(=O)CC(O)c2ccccc2)CC)OCCC1(C)C 74799,C1(N(C(c2n[nH]c(C)n2)=O)CC)CCN(C(c2cc(OC)c(Br)s2)=O)CC1 74800,c1(C(C)C)ncncc1C(=O)NC1CN(C(=O)C(O)CN(C)C)CC1C 74801,N1(C(C(c2ccn(C)c2)C)=O)CCC(C(=O)NC2CC23CCCCC3)C(O)C1 74802,CN1CCn2ncc(C(N3CC4(C3)CN(C(c3nnn(C)c3N)=O)C4)=O)c2C1 74803,C1(C(N(CC(=O)N(CC)CC)C)=O)CC(NC(=O)CCc2cnco2)C1(C)C 74804,N1(C(C(F)=C(C)C)=O)CCC(C)C1CNC(=O)COc1ccccc1F 74805,c1(N2CCC(N(C)C(C3CCc4nnnn4CC3)=O)C2)c(Cl)cncc1[N+](=O)[O-] 74806,Cc1ccnc2c(C(=O)NC(C)CNC(=O)CNC(=O)CC(F)(F)F)cccc12 74807,CC1=C(CNC(c2ccc(C(C)(C)C)cc2O)=O)SCCO1 74808,N1(CC(C)(O)C2CC2)CCCC1c1ccc(Br)s1.CNC 74809,c1(NC(C(n2c(-c3ccccc3)cc(C)n2)CCl)=O)ccc2ncnn2c1 74810,C1(NC(c2ccc(C(F)(F)F)nc2)=O)CCN(C(C2CCCOCC2)=O)CC1F 74811,N1(C(CC(C)C)=O)CCC2(CCCCN(C(=O)C(O)C(F)F)C2)C1 74812,N1(C(Cn2ccc(C)n2)=O)CCCC(C(=O)NCC2CC23CC3(F)F)(CO)C1 74813,CC(Cc1cnco1)C(=O)N(CCNC(=O)C(F)C1CCC1)CC1CC1 74814,C1(CCC)CN(C(c2ncoc2-c2ccc(OC(F)(F)F)cc2)=O)CCO1 74815,c1(CC)ccccc1NC(=O)CN(C(=O)CC1CC(C)OC1C)C(C)C 74816,Cc1oc(C)c(C(=O)NC2CCOCC2NC(C2CC2F)=O)c1C 74817,N1(C(c2cn(CC)nc2)=O)CCC(NC(=O)C2=CC(O)CCC2)C(C)(C)C1 74818,N1(C(C(C)N2CCC2)=O)CC2(CCCC2NC(=O)CC2CCC3CC23)C1 74819,N1(C(C(F)=CC)=O)CCN(C(c2ccccc2-c2nc(C)no2)=O)C(CCO)C1 74820,c1(C(=O)NC(C2CCN(C(=O)CC3NC(=O)NC3=O)C2)C)cc(Cl)nc(=N)[nH]1 74821,C(CC1(C)CC1)(C(=O)NCC1CCC1)N(C(C)C)C1CC1 74822,C1(NC(c2c(C)ccc(C)n2)=O)CC2CC(C1)N(C(c1ccc(=O)oc1)=O)C2 74823,C1(CNC(c2c(C)cncn2)=O)CN(C(C23CC(C)(CCO2)C3)=O)CCC1C 74824,c1(C(=O)NC23CCCC(NC(c4sccc4F)=O)(C2)C3)cc2n(n1)CCCC2 74825,c1(CCNCC(C2CCCOC2)OC)cn(C)c2cc(Cl)ccc12 74826,N1(C(C(CCC)NC(=O)CCn2ccnn2)=O)CC2CC1C1CC21 74827,CCCC(CNC(=O)CC1CCCOC1)NC(c1ccoc1CC)=O 74828,C1(CNC(C(F)OC)=O)CN(C(c2cnn(C3CCCC3)c2)=O)CCC12CCC2 74829,CON(C)CCNC(=O)C(C1CCN(C(=O)CN2CSCC2=O)C1)C 74830,C(C(C)C(C)C(=O)N1CC(n2cc(-c3ccc(Cl)c(C)c3)nn2)C(C)C1)OC 74831,C12(C(=O)NCC3(OCC)CN(C)C3)CCC(CC1NC(=O)CN1CCCC1C)C2 74832,C(=O)(C(C)(C)C(C)NC(=O)C(C)=C1CCC1)N1CCC(N(C(C=CC)=O)CC)C1 74833,c1(C(=O)NC2CC3CC(NC(C(CCCOC)C)=O)CC32)cccc(F)c1C#N 74834,Cn1cc2c(n1)CCC(COC(C1CCCC(CC(N)=O)C1)=O)C2 74835,CN1CCOC(C(=O)N(C2CN(C(c3coc(CC4CC4)n3)=O)C2)C)C1 74836,C(=O)(C1OCCn2ccnc21)NCC(C)NC(c1cn(CCC2CC2)nn1)=O 74837,N1(C(CCC(=C)Cl)=O)CCC2(C1)CN(C(C1CCCC(C)O1)=O)CCO2 74838,c1(OC)cc(-c2cnc(OC)cc2C(=O)Nc2ccc(C)cc2)cc(F)c1F 74839,N1(Cc2ncc(OC)nc2)CCN(C(=O)C=Cc2ccc([N+](=O)[O-])o2)C2(CC2)C1 74840,N1(C(C(C)NC=O)=O)CC(C(N2CCC3(CCSC3)C2)=O)CCC1(C)C 74841,C(=O)(C(O)CC(C)(C)C)N1CC(C)C(NC(=O)C(C)Cn2ccnc2)C1 74842,c1(CC)ccc(F)c(C(N2CCCC(F)(CNC(c3ncc[nH]c3=O)=O)C2)=O)c1 74843,C1(CC(NOC(C)C)=O)CN(C(c2csc(F)c2)=O)C(C)(C)C1 74844,C1(OC)CC2(C1)CC(C(N1CC(NC(=O)C=CC3CC3)C(F)C1)=O)C2 74845,C(=O)(CC1=CCCCC1)NC1(COC)CN(C(C2CC(C)CC(C)C2)=O)C1 74846,Cc1ocnc1CC(=O)NCC(c1ccccc1)CNC(C1CC(C)(C)C1)=O 74847,CC(C)(F)C(=O)N1CCCC1C1(O)CN(C(=O)CSCC2CCCCO2)C1 74848,c1(OC)cccc(C(N2CCC(C)C(NC(=O)C(F)C(F)(F)F)C2)=O)c1F 74849,C1(NC(c2n[nH]c(C)c2C)=O)CCCC12CN(C(=O)C#CC(C)(C)O)C2 74850,CN1C2CCC1CC(=CC(N1CCC(NC(=O)C(N)=O)C(CO)CC1)=O)C2 74851,Cc1cc(CCC(=O)NCCC(C)NC(c2cccc(CS(C)=O)c2)=O)c(C)o1 74852,CC1CCC(CNC(c2cc(Cl)c(Cl)s2)=O)N(C(c2cnn(C)n2)=O)C1 74853,N1(C(CC(CC)C)=O)CCCC2(COCC(=O)N2)C1 74854,CC(C)(COCC(F)F)C(=O)N1CCOC(CNC(=O)CC2CC3(CC3)CO2)C1 74855,N1(C(c2ccc(SC)s2)=O)C2CCC1CC(N(C(=O)Cn1ccc(C)n1)C)C2 74856,C1(C(=O)NC(C=C)COC)(CNC(C2CCC(C)O2)=O)CC(C)(C)C1 74857,C1(C(=O)NC(C(=O)NCCCc2cnccn2)C2(C)CC2)CC2C(C1)C2(C)C 74858,N1(C(c2cc(C#C)cc(F)c2)=O)CCC(C2CCN(C(=O)CC3CC3)CC2)CC1 74859,c1(CC(=O)NC23CC(C(N(C(C)(C)C)CCN)=O)(C2)C3)cc(F)cc(Br)c1 74860,c1(CNC(c2cnns2)=O)ccc(CCNC(C2CCO2)=O)cc1 74861,Cc1ccnn1C(C)C(N1CCCC1C1(C(=O)NC2(C(C)C)CC2)CC1)=O 74862,N1(C(COCCC=C)=O)CCC(CCNC(=O)C(C(C)O)N(C)C)CC1 74863,c1(C(=O)NC2CC3CN(C(c4c(OC)ccs4)=O)CC32)csc2c1CCC(C)C2 74864,C1(C(N(C(C)CNC(=O)Cc2nc(C)c(C)o2)CC)=O)CCC2(CCC2)CO1 74865,N1(C(CC2N(C(=O)CC3C=CCCC3)CC(F)C2)=O)CCC12CCSCC2 74866,CC1(CNC(=O)CN2CCCC(C(F)(F)F)C2=O)CCCN(C(=O)C(N)=O)C1 74867,CCC(O)C(F)(F)C(=O)NCC(C)(C)CNC(C1CC(=O)N(c2nccs2)C1)=O 74868,C1(C(=O)NCC(COC)NC(c2csc(C)c2C)=O)CCCCC(=O)N1 74869,N1(C(c2n(CCC)ncc2)=O)CCC2(CCC2)C(CNC(C2CSC2)=O)C1 74870,N1(C(C(C)(C)OCC)=O)CC2COCC2(C(=O)N(C)CC2(COC)CC2)C1 74871,Cc1noc(C)c1CC(=O)NCC(C)(C(C)C)NC(=O)CC1CC(F)(F)C1 74872,CC(C(=O)NC(=O)C1=CCNC1)S(=O)(=O)NC1CC1 74873,C1(C(=O)Nc2c(C)nn(CCF)c2)CCCCN(C(C2CCC3(CCC3)O2)=O)C1 74874,N1(C(C2C(=C)C2)=O)CCC(CNC(c2cccc(C3CC(OC)C3)c2)=O)C12CC2 74875,C1(NC(C=NOC)=O)CCCC(CNC(=O)CNc2ccnc(C(F)(F)F)c2)C1 74876,C1(C(=O)NCC2(OC)CCN(C(c3c(C)nsc3C)=O)C2)CC(S(C)(=O)=O)C1 74877,CC1(C)CCN(C(=O)Nc2cccc(CNC(=O)OC(C)(C)C)c2)CC1 74878,C1(CCC)CCCN1C(=O)COc1nncs1 74879,c1(OCCNC(N(C(CSC)Cc2cccs2)C)=O)ccccc1 74880,N1(c2ncc(C(=O)OC)cn2)CC2CCC1C(NC(C1CCN(C)C(=O)C1)=O)C2 74881,C1(CNC(C=C(C)Cl)=O)CN(C(=O)C(c2ccc(F)c(Cl)c2)C)CC(C)(C)O1 74882,CC(C(=O)NCC(C1CCCC1)NC(c1nccs1)=O)C1CCCC1 74883,N(C(=NCCn1cccn1)NCCN1CCCC1)C(c1ncccc1Br)C 74884,N1(C(C2CN(C(N)=O)C2)=O)CCCC2C1CCCCN2C(c1cc(Cl)c[nH]1)=O 74885,N1(C(COCc2onc(CC)n2)=O)CCC2CCN(C(=O)CC(C)(F)F)CC12 74886,CCCC(C)(O)CC(=O)NCC1(OC)CCN(C(C2CCCCN2C(N)=O)=O)C1 74887,c1(-n2c(Cc3cn(C(C)C)nc3)nc(C3CC3)n2)ccc(S(C)(=O)=O)cc1 74888,CC1CCC(NC(=O)CCc2cnccn2)CN1C(c1cc(Cl)cnn1)=O 74889,c1(C(=O)NC2C(NC(c3ccc(CC)o3)=O)CCOC2)ccnc(OC)c1F 74890,C1(C(N2CCC(CCNC(CSCCC(C)C)=O)C2)=O)CC2CCC(C1)C2F 74891,C1(CC)(NC(c2ccc(F)cc2Cl)=O)CCCN(C(=O)C(O)CCSC)C1 74892,N1(C(C(C2CC2)OCC)=O)CCN(C(c2ccc(CC)[nH]2)=O)C(C2CCCC2)C1 74893,c1(CN(CC(COCC)O)C)ccc(C(F)(F)F)c2c1OCCO2 74894,Cc1cc(C)c(C(=O)N(CC(O)CNC(c2ccc(C(C)(C)C)nc2)=O)C)s1 74895,c1(C(=O)NCCC(C)NC(CCCNC(C)=O)=O)c[nH]c2ncccc12 74896,N1(C(CC(C)N2CCCC2=O)=O)CCN(C(C2C3CC4C(C3=O)C24)=O)CC1CO 74897,Cc1cc(C=CC(=O)NCCC2CCN(C(=O)Cn3cc(Cl)cn3)C2)on1 74898,C1(CNC(CCSC)=O)CCC(C)CN1C(c1cc(C(N)=O)c[nH]1)=O 74899,N1(C(CCN(C(=O)CC2CC2)C2CCC2)=O)CCN2CCC1CC2 74900,S(=O)(=O)(c1ccc(N2CCC(CC)(CC)C2)nc1)N(CCC)Cc1ccc(Cl)s1 74901,C12(C(=O)NCCC3N(C(c4ncc(OC)cn4)=O)CCCC3)CCCC1C2(F)F 74902,c1(OCC(=O)NCCCCN(C(C(C)OCC(C)C)=O)C)ccc(F)cn1 74903,N1(C(C(CCSC)NC(=O)CN2CCCCC2C)=O)CCCC(C)C1CO 74904,C=CC(C)(O)CC(=O)N1CCCCC(C(N2CCC(OC3CC3)C2)=O)C1 74905,CC1CCN(CC(=O)N(C2CCC(NC(=O)C3=C(Cl)CC3)C2)C)CC1 74906,c1(C(C(=O)NC(C)(C)CC)N(CC=C)C)cc(C2CCC2)[nH]n1.C(COC)SC 74907,c1(C2(C(=O)NC(CNC(C3(OC)CCSC3)=O)C(C)C)CC2)ccc(Cl)c(F)c1 74908,C1(C(C)NC(CC=C)=O)CN(C(=O)CCC2CCC(=O)N2)CCO1 74909,c1(CCCNC2CC(OCC)C2=Cc2ccccc2)cc(O)n(C)n1 74910,N1(C(c2ccc(NS(C)(=O)=O)cc2)=O)CCN(C(C2CCOC2)=O)C(CCO)C1 74911,C1(C)(C(=O)NC2CCC(NC(CCCCCOCC)=O)CC2)CC(C2CC2)=NO1 74912,CC1CN(C(=O)C=Cc2cncs2)CC1n1cc(COCCOCCO)nn1 74913,N1(C(CCCOCCC)=O)CCN(C)CC1CNC(c1ccc(CC)s1)=O 74914,c1(CC)cccnc1C(=O)NC1(C(N2CCN(CCO)CC2)=O)CC(F)(F)C1 74915,C1(CNC(c2cccnc2)=O)CCN(C(=O)CC(O)C2CC2)C1 74916,Cc1nnn(CC(=O)NC2CCCC2CN(C)C(c2cc[nH]n2)=O)n1 74917,c1(NCCC2CCCN(NC(=O)OC(C)(C)C)CC2)nc2c(cc1Cl)C(=O)OC2 74918,C1(C(N2CCC(C(C)NC(c3cnn(C4CCC4)c3)=O)C2)=O)CC2CC2CC1C 74919,c1(N2CC(C)=C(C)C2)nc(=NCCC2CCN(C)CC2)[nH]c2c1COCC2 74920,C1(C(N(C(C)Cc2cccs2)C)=O)CCCC1c1nc[nH]n1 74921,C12(C(N3CCCC(C(=O)NC4CC5CCC4O5)C3)=O)CCC(CC1)CC2 74922,N1(C(c2ccc(CCCC#N)cc2)=O)CC2(CO)CCCC2(F)C1 74923,c1(OCC(=O)NCC2(NC(c3c(CC)con3)=O)CCC2)c(Cl)cccc1Cl 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75210,Cc1nc(C(=O)N(C(c2ccccc2)CNC(=O)CCCC#N)C)cn1C 75211,C1(C(=O)NCC2(C(N)=O)CN(C(CC(CC)C3CC3)=O)C2)CC2CCC(C1)C2=O 75212,C(=O)(C(CC(=O)NC1(CNC(c2cc3oc(C)cc3[nH]2)=O)CC1)C(C)=O)OCC 75213,N1(C(Cn2c(C)nnn2)=O)CCC2(C1)CN(C(C1(O)CC(C)(C)C1)=O)C2 75214,c1(CNC(C(CCC#C)O)=O)nn(C)c2c1CN(C(=O)C(C)N(C)C(C)=O)CC2 75215,Cc1nc(Br)c(Br)n1CC(=O)NC(c1ccnn1C)CO 75216,C1(C(N(CC(CN(C(C2(OCC)CC2)=O)C)O)C)=O)CN2CCCN1CC2 75217,c1(NC(N2C(C(=O)OC)C(C)CC2)=O)cc(C)cnc1OC 75218,c1(C(=O)NC(CNC(CC(n2c(CC)ncc2)C)=O)CO)sc(C)c(C)c1C 75219,CCC(C)C(O)C(C)C(=O)NC(C(=O)NCCc1ccncc1C)c1cccs1 75220,C(C)(CO)(C(=O)NC(C1(O)CN(C(c2ccc(CC(C)C)s2)=O)C1)C)OC 75221,c1(C(=O)NCC(CN(C(C2CCS(=O)(=O)C2)=O)CC)(C)C)ccccc1C 75222,C(=O)(C(F)(F)CCn1cccn1)NCCOC1CC(NC(=O)CC(F)(F)F)C1 75223,N1(C(c2cc(C)ncn2)=O)CCC(CNC(C2COC(=O)N2)=O)C1(C)C 75224,C(CCC(C(=O)N(C(C)CC1CC1)C)NC(=O)CC1CCCC(=O)N1)OC 75225,C1(NC(c2c(C)cn(C)c2)=O)C(C)CCN(c2ncns2)C1C 75226,N1(C(c2cc(C)cc(F)c2)=O)CCCN(C(C2CC=CCC2C)=O)CC1CO 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75244,N1(C(c2ccc(F)s2)C(=O)NCC)CCc2c(cc(F)c(F)c2F)C1 75245,c1(C(=O)NCC2N(C(C(C(C)C)C3CCC3)=O)CC(O)C2)ccn2ncnc2c1 75246,Cc1ccc(C#N)cc1C(N1CC(C)(CCC(=O)N(CCCO)CCCO)C1)=O 75247,c1(C(N2CCC(O)(CN(C(C3CCC(=C)CC3)=O)C)C2)=O)cc2ccsc2n1C 75248,C1(O)(CNC(c2cn(CC(C)C)nc2)=O)CCCN(C(C2(C)CC2(F)F)=O)CC1 75249,C123C(C4CC1C2C4)N3.c1(CN(CCCOC)C(=O)OC(C)(C)C)cccs1 75250,Cc1c(C(=O)NCC2CN(C(c3occ4c3CCC4)=O)CC2C)cncc1Cl 75251,c1(C(=O)NCCC(CNC(c2c(C)n(C)nn2)=O)O)cc(C(F)(F)F)ccc1F 75252,c1(N2CC(CO)OCC2)nc(N2CC=C(c3cccs3)C2)nc2ccccc12 75253,n1(C(C)C)cnc2c(NCC3(C)CS(=O)(=O)C3)[nH]c(=NC3CCCCC3C)nc12 75254,C1(S(C)=O)(C(=O)OC)CCN(C(c2c(Br)nc3n2CCOC3)=O)CC1 75255,Cn1c(=O)n(CC(N2CCC(CC(=O)Nc3nccs3)C2)=O)c2ccccc12 75256,C(CNC(c1cocn1)=O)(CC(F)(F)F)NC(CN1CCCC(CC)C1)=O 75257,c1(CC)c(C(=O)NC2CC(NC(=O)C(F)CC)C(O)C2)csc1C 75258,c1(C(=O)OC)nc(Cl)cc(=NC2CC3CN(C(c4ccc5c(c4)CC5)=O)CC23)[nH]1 75259,C1(NC(c2c(C)n[nH]c2)=O)CCCN(C(=O)CCCC(C)N2CCOCC2)C1C 75260,O=C(C1CCc2ccccc21)NCC1CCCC1NC(C1CCCS1(=O)=O)=O 75261,c1(C(N2C(CNC(CC(C(=C)C)O)=O)CC2)=O)ccsc1S(N)(=O)=O 75262,N1(C2CC3N(C(c4ccc(C)c(C)c4)=O)C(CC3)C2)CCCC(F)C(F)(F)C1 75263,c1(C(N(CC(C)NC(=O)NN2CC3CCC2C3)CC)=O)cc(CO)cc(CC)c1 75264,C1(C(N2CC(OCCCCC)C2)=O)C=CCN1C(=O)C(n1ccc(C)n1)C 75265,C1(NC(c2ccc(C(CC)C)cc2)=O)CCN(C(=O)C(C)C(C)C)C12CCC2 75266,C1(OC)CN(C(=O)CC2(O)CCCC2)CC1NC(=O)C(C)Sc1ccccc1 75267,CCC(C(=O)NCC(C)NC(C1CN(S(C)(=O)=O)C1)=O)n1nccc1C 75268,N1(C(c2c(CC)ccs2)=O)CCC(C(N2CCCCCC2)=O)C1C(C)C 75269,c1(C(=O)NC(C(C)NC(CS(CC)=O)=O)(C)C)cc(F)c(C#N)c(F)c1 75270,C=C(Cl)C(C)(C)C(=O)N1CCC(C)(CNC(c2c[nH]c(-c3ccncc3)n2)=O)C1 75271,c1(C(=O)NC2C(NC(CCSC)=O)CS(=O)(=O)C2)ccc2ncn(C)c2n1 75272,C1(CC)CN(C(=O)CCCN(C)C)CCC1NC(C1(F)CCCC1)=O 75273,C1(CCNC(COCC(=C)C)=O)CN(C(c2cnc(N(C)C)s2)=O)CCO1 75274,N1(C(c2ccnc3[nH]nnc23)=O)CCC2CCC(C1)N2C(C1CC=CCC1)=O 75275,N1(C(c2cc(OC)ns2)C(=O)NCCCC2CC2)CCCc2c(C)cccc21 75276,C(C(C)(C)CCC#N)(c1nnnn1C)NCc1n(CCC)ncn1 75277,n1(CCC)ncc(C(=O)NC2C3CC(NC(c4nocc4C(C)C)=O)CC23)c1C 75278,C1(CC=C)(NC(C2CCCO2)=O)CCN(C(c2ccc(N)c(Br)n2)=O)CC1 75279,C(=O)(CC(F)(F)C(F)F)NC(CC(C)NC(c1c(C)nc(C2CCCC2)s1)=O)C 75280,C1(C(=O)NC(c2nc[nH]n2)C)(CNC(c2nonc2N)=O)CCCCC1 75281,C(=O)(CC(C(F)F)c1ccc(F)cc1C)N(C1CN(C(=O)C2CC2)CC12CC2)C 75282,n1(CCCC)nc(C)c(C=CC(=O)N(CC(C)(C)NC(=O)CC(C)(C)O)C)c1Cl 75283,C(c1ccc(OC(F)F)cc1)=CC(=O)NCCn1ccnc1.C=CC 75284,N1(C(C(CC)CC2CCCCC2)=O)CC(C)(CNC(C2(O)CC2)=O)CC1(C)C 75285,C1(C(=O)NCC2CC(C(=O)OC)C2)CC12CCN(C(=O)C1=CCN(C)C1)C2 75286,N1(C(CC(C#C)O)=O)CC(C)(C)CC(C)(C)C1 75287,C1(F)(C(=O)NCCc2c(CNC(CC(C)OC)=O)nco2)CCS(=O)(=O)C1 75288,C1(CNC(C(C=C)O)=O)CCN(C(c2nc(OC)c(C)s2)=O)C1(C)C 75289,N1(C(CCC)C)CC(C(=O)NCCCCCCNC(=O)C2=CCC2)CC1=O 75290,CCCC(C(C)(C)C)NC(=O)CCC1CCN(C(=O)Cc2csnn2)CC1 75291,N1(C(C)C)CC(C(=O)N(C)CC2(NC(C3CC(CF)C3)=O)CC2)CCC1=O 75292,C1(CC(=O)NC2CCCC2NC(C2CC3CCC2C3)=O)CCC(F)(F)CC1 75293,c1(NC2C(CNC(C3(OC)CCCOC3)=O)CCCC2)ncc(Cl)cc1[N+](=O)[O-] 75294,N1(C(C(C=C)OC)=O)CC(O)CC1C(=O)NCCOC1CCOC1 75295,N1(C(c2ccoc2Cl)=O)CCCC1C1CCCN1C(c1c[nH]nc1Br)=O 75296,c1(C(N(C(C(N2CCC(OC(C)C)C2)=O)(C)C2CC2)C)=O)c[nH]c(=S)cn1 75297,C=CCC(CC(=O)NC(C)C(=O)NC1CC1)NC(=O)COC1CCOC1 75298,C(=O)(CC(c1ccccc1)NC(C1CCCN1C(N)=O)=O)N(C)CC1CC12CC2 75299,c1(C(N2CC(O)(CNC(C3N(C(CC)=O)CCCC3)=O)C2)=O)cc(N)ccc1O 75300,c1(C(=O)NCC(C)N(C(=O)CCc2cncn2C)CC)cc(F)cnc1O 75301,Cc1cnc(C)c(NC(c2c(NC(c3ccc(O)cc3Br)=O)cccc2F)=O)n1 75302,c1(-c2nc(C3(CO)CCN(C(=O)OC(C)(C)C)C3)on2)cccc2c1CCCC2 75303,C(=O)(CC1=NNC(=O)C1)NC1CCN(C(c2n(CCCC)ncc2)=O)CC1F 75304,C1(NC(=O)CSc2nnc(S)s2)C2CC1CN(C(=O)CSc1ccccn1)C2 75305,N1(C(C(F)OC)=O)CCCC1CN(C(=O)C(C)(C)N(S(C)(=O)=O)C)C 75306,C(C(C)(C)S(C)(=O)=O)CCN(c1ccc(C(F)(F)Cl)cc1)C 75307,CC(C)(C#Cc1cn(Cc2cncs2)nn1)NC(=O)Cc1ncccc1Br 75308,N1(C(c2c(OC)c[nH]n2)=O)CCN(C(c2ccc(F)cn2)=O)C(c2ncc[nH]2)C1 75309,C1(CC(=O)NCC(COC)C)CC2(C1)CN(C(=O)C(C)C(F)(F)F)C2 75310,c1(C(=O)NCC23CC2CN(C(=O)C(=Cc2c[nH]cn2)F)C3)nsc2ccccc12 75311,C1(F)(CNC(C(CC(C)C)N(C)C)=O)CCCN(C(=O)OC(C)(C)C)CC1 75312,N1(C(c2cn(CC=C)nn2)=O)CCC(F)C(NC(c2cc(C3(C)CC3)n[nH]2)=O)C1 75313,CCC(C)(CN=c1ccnc(N2CCCC(C3CCC3)CC2)[nH]1)c1ccncc1 75314,c1(OCCC)cccc(CN(C=O)C(c2ccncc2)c2cc(C)no2)c1 75315,c1(C(=O)NCC2CC(CC)CN2C(c2cc(=O)n(C)cn2)=O)ccc(F)c(O)c1 75316,CCCCC(CNC(C1C2CCC12)=O)NC(=O)CCCNC(=O)NC 75317,Cn1cc(C(C(=O)NCCC(C)(C)O)NC(=O)CNC(N)=O)nn1 75318,c1(NCC)cc(Cl)ccc1C(N1CCCC(O)(CNC(=O)C=CSC)C1)=O 75319,N1(C(=O)CC2=CCCC2)CCOC2(CCN(Cc3cc4cnccc4[nH]3)CC2)C1 75320,CCC(CC)C(C)NC(C1OCCC1NC(=O)C(C)(C1(C)CC1)OC)=O 75321,Cn1ncc([N+](=O)[O-])c1C(=O)NC1CCCC(NC(=O)C=CCF)CC1 75322,c1(C(=O)NCCC(C(C)C)NC(c2c(CC)nc[nH]2)=O)cccc2oc(O)nc12 75323,c1(OCC2CC(NC(CCn3cc(CCCC(C)O)nn3)=O)C2)ccc(F)cc1 75324,CCCC(O)C(=O)N1CCC(C2N(C(=O)C=CC3CC3)CC2(C)C)CC1 75325,C1(C(=O)NCC2(C(=O)N(C3CCCC(O)C3)C)CC(=C)C2)CCN(C)C1=O 75326,C1(C)(COC)C=CCCN1Cc1cccnc1-c1ccc(Cl)cc1.C1C(=O)N1 75327,c1(CC)cc(C(N2CCOCC2CC(=O)NC(C)Cc2cnc[nH]2)=O)ncn1 75328,C(C(C)C(C)C(=O)NC(C1(O)CN(C(=O)C(O)C2CCC2)C1)C)OC 75329,C1(NC(C2(CC(C)C)CCCC2)=O)CC2CC(NC(c3ccc(Cl)cn3)=O)C2C1 75330,c1(C(=O)NCC2CCN(C(c3cnc(CC)[nH]3)=O)C2)c(C)cc(C)nc1O 75331,Cc1cc(N)c(C(=O)NCC23CCCC2CCN3C(c2ocnc2C)=O)nc1C 75332,O=C(C#CC1CC1)NCC12CC1CN(C(C1CC(=O)N(CC3CC3)C1)=O)C2 75333,N1(C(C)=O)CC(NC(C=CC(=O)NCC2(COC)CC(F)(F)C2)=O)CC1(C)C 75334,c1(C(=O)NCC(C)N(C)C(c2ncncc2Cl)=O)c[nH]cc(Cl)c1=O 75335,CC1CC(=O)NCC1C(N1CCCC1(C)CNC(C1CC(O)C1)=O)=O 75336,c1(OC)ccc(Br)nc1CN1CCCC(C)(C(=O)Nc2nc(Br)ccc2Br)C1 75337,Cc1cnoc1C(=O)N(C(C)CNC(=O)CC1(N2CCOCC2)CC1)CCO 75338,C#CCC(C)(CC)C(=O)NC1C2CC3C1C3C2C(=O)NCC(C#C)OC 75339,CCCCCCCCC(=O)N(C1CCCN(C(=O)CC2CCCCC2O)C1)C 75340,CCCC(CCC)=CC(=O)N(CC)Cc1cn(-c2cc(C)nn2C)nn1 75341,C1(C(N2C(C)CCC2C(=O)Nc2ccc(F)nc2)=O)CC2CCCC2C1 75342,c1(C(=O)NCCCN(C(C(CC)OC)=O)C2CCCC2)ccc(C)n1C 75343,c1(COC)ccsc1C(=O)N(C1CCN(C(=O)CCC=C(C)C)C1)CCO 75344,C12(C(N3C(CNC(=O)C4=CCCCC4)CCC3)=O)CC1COC21CCC1 75345,CC1(C)C(C)(C(=O)NCC2(O)CN(C(c3ccccc3CC#N)=O)C2)C1(C)C 75346,c1(C(C)=O)ccc(C(=O)NC(c2ccccc2)CNC(=O)C(C)CC2CCC2)s1 75347,C(C(=O)NNC(=O)C1=CS(=O)CCC1)(c1ccccc1)OC 75348,Cc1cc(C(=O)NC2CC(CNC(=O)CN(C3CCCC3)C)C2(C)C)cn1C 75349,C(=O)(CC(C)(C(F)F)N(C)C)N1CCN(C(c2c(C)[nH]c(C#N)c2)=O)CC1CO 75350,N1(C(CC(=O)NCC)=O)CCN(C(C)CNC(c2cnns2)=O)CC1 75351,c1(C(N2C(C)CC(NC(=O)Cc3ccco3)C2)=O)cc(C(F)F)ccc1Cl 75352,N1(C(c2nc(C)c(C)s2)C(=O)NCC)CC(C)C(C)C1C 75353,c1(N(CC)CC)ccc(CCC(=O)NCC(CC)NC(C2CCC2(C)C)=O)cc1 75354,CC(C(=O)N1CCC(N2CCN(C(C3CCC(=O)N3C)=O)CC2)C1)P(C)(C)=O 75355,C1(C(=O)NC2CC(CNC(c3ccsc3C)=O)C2)(OCC)CCSCC1 75356,C1(F)CCN(C)C1.C1(C(C)C(=O)N)CCN(C(=O)CCc2cscn2)CC1 75357,Cc1cc2[nH]c(C(=O)NC3CC4(CCN(C(C56CC(CO5)C6)=O)C4)C3)cc2o1 75358,N1(C(C2(CNC(c3cnn(C)n3)=O)CCCCC2)=O)CC(O)C(O)C12CCC2 75359,C(C)(C)(CC(=O)NCc1ccoc1C(=O)NCCCC(O)CO)N(C)C 75360,c1(C(C(=O)NC(C)C(=O)OC)N(CCCC)C)cc(OC)c(Br)cc1F 75361,N1(C(CC2CCCN(C(C=CCC)=O)CC2)=O)CC2CCCC2C12CC2 75362,CC1CCN(C(c2ccc3c[nH]nc3c2)=O)C(C)C1NC(c1ccc(F)nc1)=O 75363,C1(NC(c2cc(C)nc(C)n2)=O)CC2CCC(C1)N2C(=O)C(O)c1cnc[nH]1 75364,c1(C(=O)NC2CCC(F)(SC(C)C)C2)ccc(NC(c2ccncc2)=O)cc1Cl 75365,c1(OC)cccc2[nH]c(CN3CC(C(N4CC(F)C(F)C4)=O)CC(F)(F)C3)cc12 75366,C(=O)(C(F)(F)C(C)(C)O)N1CC(C)CC(C(=O)NC2CCC(C(C)C)CC2)C1 75367,CCC(O)C(F)(F)C(=O)NCCCC1CCN(C(=O)CC(C)C(C)(C)C)CC1 75368,N1(C(CC=C)=O)CCC2(CO)CN(C(c3coc4cc(F)cc(F)c34)=O)CC2C1 75369,Cc1cc(C)c(C(=O)NCCN(C(=O)CC2CC2C)C)c(C)c1 75370,N1(C(C(CCN(C)C)NC(=O)CCn2ccnc2)=O)CCC(F)(F)C(F)C1 75371,C#Cc1ccc(OCC(=O)NCC2CCN(C(=O)C(CC)CC=C)CC2O)cc1 75372,O=C(C1CCc2ccccc21)NC1CN(C(C2CCC(C(=O)O)CC2)=O)CC1F 75373,CN=c1nc(N2CCOc3cccc(Cl)c3C2)[nH]c(=NC(C)C2CCN(C)C2)[nH]1 75374,C1(N(C(=O)Cc2ccsc2Cl)C)CC2CC1N(C(c1ccncc1F)=O)C2 75375,C1(C(=O)NC(CN(C(=O)COC(F)F)C)CO)Cc2cccc(OC(F)F)c2O1 75376,C(=O)(CCCC(F)(F)F)N1C(CNC(C2C(C)C2)=O)COCC1 75377,c1(C(N2CCN(C(CN(CC)CC)=O)C(C3CC3)C2)=O)cnc2n1CCC(C)C2 75378,C1(C)(C(=O)Nc2c(C(=O)OC)n[nH]c2)COCCN1C(C1NC(=O)NC1=O)=O 75379,Cc1ccc(C(=O)NCC2(NC(C3CCCCN3C)=O)CCCCC2C)c(N)c1 75380,N1(S(CC#N)(=O)=O)CCc2cccc(C(N3CC4C(C3)C4(C)C)=O)c2C1 75381,C1(C)(CC(=O)NC(COCC)C)CCN1C(=O)CC1(C)OCCO1 75382,C1(C(N2CCC(C(C)NC(c3cscn3)=O)C2)=O)CC1C1CC1C 75383,N1(C(c2ccccc2Cl)C(=O)NCC)CCn2c(CC)nnc2C1 75384,Cc1ccc(Cl)cc1-c1cn(CCCN(C)C(c2csc(CO)n2)=O)nn1 75385,CC1(C)CCCCC1C(=O)NC1C=CC(C(=O)NCC2CC(O)C(O)C2)C1 75386,N1(C(c2cc(C)on2)=O)CCC(F)(C(=O)NC(C2CCCOC2)(C)C)CC1 75387,N1(C(C(N2CCOCC2)C)=O)CC(NC(c2sc(Cl)cc2Cl)=O)CC1(C)C 75388,N1(C(C2(S(N)(=O)=O)CC2)=O)CCC2(C1)CN(C(=O)CC1COC3(CCC3)CO1)C2 75389,C1(CC(=O)N(CCNC(c2cscc2Br)=O)CC)CC(C)(C)OC1=O 75390,C(C(C)(C)CC(=O)NCC(C1CC1)NC(C1CC(C)(C)CO1)=O)N(C)C 75391,c1(C(=O)NCC2CC(NC(C34CCC(CC3)OC4)=O)C2)cc2cc(Cl)ccc2o1 75392,C1(O)(CNC(C2(CSC)CCC2)=O)CCN(C(=O)Cc2ccc(O)cc2Cl)CC1 75393,N1(C(CN(C)C(N)=O)=O)CCCC2CN(C(=O)CCc3cnn(C)c3)CCCC12 75394,c1(C(N2CC(CC)C(NC(c3ccncc3)=O)CC2)=O)cc2nc(Cl)ccc2s1 75395,C1(C(=O)NC(CCC)(C)CC)CCC2(CC2)N1C(C1CCCOCC1)=O 75396,c1(CC)ncccc1C(N1CCCC1C(C)NC(c1ccnnc1)=O)=O 75397,N1(C(c2c(C)cnnc2)=O)CCc2cccc(C(N3CCSCC3)=O)c2C1 75398,C1(C(=O)NCc2ccsn2)CN(C(=O)C(c2cccc(Br)c2)O)CCC1(F)F 75399,CC1CC(CN2CCCC2Cc2ccncc2)CCO1 75400,CCCCC(O)CC(=O)NCC1(O)CC(NC(=O)CCOc2ccc(C)cc2)C1 75401,C1(C)(NC(C=CCN(C)C)=O)CCN(C(=O)Cn2cnccc2=O)CC1 75402,c1(C(=O)NC2CC3(CN(C(CCCCC)=O)C3)C2)c(Cl)ccc(OC)c1N 75403,Cc1cc(=NCC(Cc2cccs2)C(C)C)[nH]c(=NCC(C)Cc2cn[nH]c2)[nH]1 75404,N1(C(C(C(CC)C)O)=O)CCCC2(C1)CN(C(=O)C1=NNC(C(F)(F)F)C1)C2 75405,C1(C(=O)NCC(C)N(C(=O)CCC(=O)c2ccc(F)cc2)C)CCC2CCC1O2 75406,C1(CN(C)CC2(c3ccccc3)CCCC2)CC(=O)C12CC2 75407,N1(C(C2(F)CCN(C(c3cnc(N(C)C)o3)=O)C2)=O)C2CCC1COC2 75408,Cc1cc(NC2CC(CNC(c3cc(C(N)=O)[nH]n3)=O)C2)nc(CC2CC2)n1 75409,C1(CNC(C=C(C)C2CC2)=O)(CNC(=O)C(C)NC(c2ccoc2)=O)CCCC1 75410,C1(CNC(c2cnc(C)s2)=O)CCN(C(=O)C(C2CCCCC2)O)C1(C)C 75411,c1(C(C(=O)NCCC#N)N(C(CCSC)CO)C)ccc(CF)cc1 75412,C12(C(N3CCC(COC(C)=O)C3)=O)CCCC1CCN2C(=O)C1=CC2C=CC1C2 75413,N1(C(CC(C)C)=O)CC(CO)C2(CCN(C(=O)C(C)c3ccco3)CC2)C1 75414,C1(C(=O)NCC2COCCN(C(c3cc(OC)n[nH]3)=O)C2)Cc2ccccc2O1 75415,C1(NC(c2cc(C)n(C3CCCOC3)c2C)=O)CNC(C)(C)COC1 75416,CC1CC(NC(=O)CNC(=O)OC(C)(C)C)CN(C(c2ncccc2Br)=O)C1 75417,c1(CC)cc(NC(N2CCCC2CC(c2ccccc2)O)=O)n(C)n1 75418,N1(C(c2ccc(CNC(c3occ(C(N)=O)c3)=O)o2)=O)CC(O)CC12CCC2 75419,N1(C(C(CC)n2ccnc2)=O)CCC2OCCN(C(c3nc(=O)n(C)[nH]3)=O)C2C1 75420,CC1CCCCC1C(=O)OCC(=O)NC1(C(F)(F)F)CC=CC1 75421,c1(OCC)cc(C)c(CNc2cccc(F)c2C(=O)N=c2cc(Br)[nH][nH]2)c(O)c1 75422,c1(C(N2CC(NC(C3(F)CCC3)=O)C(F)C2)=O)ccc(Br)c(Cl)c1Cl 75423,C1(S(C)(=O)=O)(C(N2CCN(C(CCSCC)=O)C(C)C2)=O)COC(=O)C1 75424,Cn1ncc(=NC(=O)C2CN(Cc3ccc4nccn4c3)CCC2O)[nH]1 75425,N1(C(c2n[nH]c(CC)c2C)=O)CCOCC(C(=O)N(CC(C)C(=O)OC)CC)C1 75426,C12(CNC(c3cn(CCOC)nc3)=O)CC1CN(C(c1ccn(CCF)n1)=O)C2 75427,C(=O)(CCC(C)(F)F)NC1(C)CC(NC(CN(C2CCC(=O)NC2)C)=O)C1 75428,C(CCOCC)(C(=O)N1CC(c2nc(=O)o[nH]2)C1)NC(C(C=C)O)=O 75429,CC1=C(C(=O)N2CCCC(C)(CNc3nnnn3-c3ccc(C)n3C)C2)CCO1 75430,Cc1ccn(CC(N2CC(CNC(c3c(C)nsc3N)=O)CC2C)=O)c(=O)c1 75431,C1(C(N2CCCC(CCNC(c3cc(C#N)sc3)=O)C2)=O)CC2C=CCC(C1)C2 75432,c1(OC)ccc2nc(C(=O)OC(C)C)c(Br)n2n1.c1(CN2CC2=O)ccccc1 75433,Cc1c(F)ccc(Cl)c1C(N1CC2CC(NC(=O)C(C)(O)C3CCC3)C2C1)=O 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75505,c1(NC(N(CCOC)C(C)C2CC2)=O)ncncc1Oc1ccsn1 75506,c1(N(C)Cc2nc(O)n[nH]2)nc(=NCc2ccsc2Cl)[nH]c2cc[nH]c12 75507,N1(C(C23CCC(F)(CC2)C3)=O)CC(NC(C2CC(n3ccnc3)C2)=O)C2(CC2)C1 75508,C1(NC(Cc2nc(CC)sc2)=O)CC2CCC1CN(C(C1CC1F)=O)C2 75509,O=[N+]([O-])c1ccn(CCSc2ccc(C(=O)NOCC=CCl)cc2)n1 75510,Cc1ccc(C(N2CCCC2(C)C(N2CC(CO)C(C)(C)C2)=O)=O)cc1O 75511,C(=O)(CCCF)N(CC(=O)NCCOC(C)(C)C)C(C)C 75512,c1(C(=O)NCCCC(=O)NC(C=C)(C)C)ccc(C#N)n1C 75513,C1(NC(N2CC([N+](=O)[O-])C2)=O)CCOC2(CCS(=O)(=O)CC2)C1 75514,CN1CCOCC1C(=O)NC1(CCC(=O)NC2(C)CC2)CCC1 75515,C1(N(CC#C)C(C2CCC(N(C)C)C2)=O)CCN(C(=O)CNC2CCCC2O)CC1 75516,c1(CCC(=O)NC(C2CCN(C(c3cnc(Cl)cn3)=O)CC2)C)ccc(=N)[nH]c1 75517,C(C(CC)(CC)C(=O)N1CCC(OCC(N)=O)C1)NC(Cc1cn(CC)nc1)=O 75518,N1(C(C(CNC(C=C(CC)CC)=O)N(C)C)=O)CCS(=O)C(C)C1 75519,c1(CC)ccc(Cl)c(C(=O)NC2CCC(NC(=O)CN(C)C)CC2)c1 75520,Cc1ccc(NC(=O)C(=O)NC(C)C)cc1NC(c1cc(Cl)sc1Cl)=O 75521,c1(CC(C)C(=O)NCCC(C)N(C(=O)CCc2ccccn2)C)ccc(F)cc1 75522,N1(C(c2n(CC)cnc2)C(=O)NC(C)C)CCS(=O)(=O)CC1 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75611,Cc1cccc(S(=O)(=O)N2CCC(NC(c3c(Cl)cccc3I)=O)C(F)C2)c1 75612,Cc1cc(C(=O)NC2CC(CCNC(=O)CNS(N)(=O)=O)C2)c(N)c(F)c1 75613,N1(C(C=CC=CC)=O)CCC(C2CC(NC(c3c[nH]c(=N)s3)=O)CCO2)CC1 75614,c1(OC)cc(C(=O)NC23CC(C2)N(C(C2(CC4CC4)CCCO2)=O)C3)ccc1Cl 75615,C(CC(C)C)(C(=O)N(C)CCN(CC)CC)NC(CC=CCCCCC)=O 75616,Cc1cccc(C)c1C(=O)NC1CCCN(C(c2cnc(C3CCC3)s2)=O)CC1 75617,C1(C(=O)OC)(SC)CC(NC(C23CC(C(C)C)(C2)C3)=O)C1 75618,CCCCCCCCC(=O)N1CC(O)(C(C)NC(=O)CCCOCCN(C)C)C1 75619,CC1(C)CCC(C)(NC(C2CCCN(C(c3[nH]nnc3C3CC3)=O)CC2)=O)C1 75620,C1(c2n(CCCSCC)nnn2)(NCCOCCN(C)C)COCCC1C 75621,c1(CNC2C=CC(C(=O)Nc3ccc(C=C)cc3)C2)ccc(F)c(C#N)c1 75622,c1(OC)ccc(CN=c2[nH]c(CC(=O)NCCN3C(=O)CSC3=S)cs2)cc1O 75623,c1(CC(N2CCC(CCC(=O)NC3CC(CC)C3)C2)=O)coc2ccccc12 75624,C(=O)(C1=CCCCO1)N(CCCC(=O)N(C(C1CCC1)C)C)C 75625,C1(NC(C2C(C=C)C2)=O)CC(C)CN(C(c2cc(C)cc(O)n2)=O)C1 75626,C(CC(C(=O)N1CCC(O)(N(C(=O)CSCCN(C)C)C)C1)N(C)C)SC 75627,c1(OC)c[nH]c(C(=O)N(C)CC2(O)CCN(C(=O)CC3CCC3(F)F)C2)cc1=O 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75645,c1(CC)cc[nH]c1C(=O)NCCOCCCN(C)C(C1(C)CC1(Cl)Cl)=O 75646,CC1(NC(C2(c3ccno3)CCC2)=O)CN(C(=O)CCc2cnoc2)C1 75647,Cc1cc2ccc(C(=O)NC3CC(C)CN(C(c4sc(C)nc4C)=O)C3)cn2c1 75648,c1(C(=O)NCC2CC(NC(=O)C(=C3CCCCC3)F)C2)cnc2ncccc2c1 75649,N1(C(C(C)(CO)NC(C2C(C=C)OCC2)=O)=O)Cc2ncsc2C1 75650,C1(NC(c2nc(Br)c[nH]2)=O)CN(C(=O)C=CCO)CC1C(F)F 75651,N1(C(CC(C)(C)F)=O)CCCC(O)(CNC(c2ccc(C(C)(F)F)cn2)=O)CC1 75652,C12(NC(C(N3C(CC)CCC3)=O)=O)CCCC1(F)CN(C(=O)Cn1cncn1)C2 75653,N1(C(C2(CCC)CC(=O)C2)=O)CCCC(C(C)C(=O)NCc2ccc(C)cc2)C1 75654,CN1CCN(CCc2nc(-c3cccs3)nn2CC2CCOCC2)CC1 75655,Cc1cccc(NNC(=O)Cn2nc(-c3ccc(F)cc3)ccc2=O)c1Cl 75656,c1(C(=O)NC2(C3N(C(C(C)OCC=C)=O)CCC3)CC2)ccc(C(C)=O)c(O)c1 75657,n1(CC(C)NC(=O)C(C)NC(=O)OC)cc(C(C)(C)NC(c2ccccc2)=O)nn1 75658,N1(C(CC(C)F)=O)CCC(C)(CNC(c2c[nH]nc2I)=O)CC1 75659,C1(N(C(=O)CS(C)(=O)=O)C)CN(C(=O)C(=O)NCC(F)(F)F)CC12CC2 75660,N1(C(=O)C=CC(c2ccccc2)=O)CC2CC1CCC2NC(=O)COC1CCC1 75661,N1(C(C2(COC)CCCCC2)=O)CC(C2CCCN(C(=O)C(C)S(N)(=O)=O)C2)C1 75662,C1(C(=O)NC2CCCN(C(C(CC)(C)C)=O)C2)(CF)CC2(CCC2)C1 75663,c1(C(=O)NCC(CNC(=O)CCc2ccoc2)F)ccn(-c2ccncc2)n1 75664,C(=O)(CCC(C)c1ccccc1)N(C1CCN(c2snc(CC)n2)C1)CC 75665,c1(N2CC(CNC(C(C)CC(N)=O)=O)OCC2)nc2c(cc1C#N)CCC2(C)C 75666,N1(C(CCC(C)OCC)=O)CC(NC(c2cc(OC)n[nH]2)=O)CC(C)C1 75667,CC1CCC(C)(C)N1C(C1CC(NC(c2csc(Cl)n2)=O)C(O)C1)=O 75668,C(=O)(CC1=NNC(=O)C1)NC1C(CNC(C(C)CC2CCC2)=O)CC1 75669,N1(C(C2C(C)CC2)=O)CCOC(C(N2CCCC2C(N)=O)=O)C1 75670,CC(C)CC(CNC(=O)C(c1cccnc1)O)NC(c1cccc(CO)c1)=O 75671,CC(C)CCN=C(NCCc1ccc(N2CCCC2)nc1)NCC1(C)CCOC1 75672,c1(C(N2CC3(CCN(C(C(C)N(CC)CC)=O)C3)C2)=O)nc2nccc(C)n2n1 75673,C(CN=c1[nH]c2c(c(=NCc3conc3C3CC3)[nH]1)CCCC2)c1nc(C)sc1 75674,c1(OC)cc(-c2ccc(-c3ccccc3)s2)nc(N2CC(CO)CC2C)n1 75675,Cc1cc(=NCC(CC(C)C)N(C)C)[nH]c(Cl)n1.N1CCCC1 75676,C1(CNC(c2oc(CC)c(C)c2)=O)COC(C)(C)CN1C(=O)CN1CCCC1=O 75677,N1(C(C2C(C)(Br)C2)C(=O)NCC2CC2)CCC23CCCCC2(C1)C3(F)F 75678,c1(C(NC(=NCCCC)NCCCC2(O)CCC2)C)ccc(S(=O)(=O)CC)cc1 75679,C1(C(N(C(C)CCNC(c2cnsc2)=O)C)=O)C2CC2CN1C(=O)OC(C)(C)C 75680,C1(CNC(c2ccon2)=O)CCC12CCN(C(=O)C(c1ccc(F)cc1)F)CC2 75681,CC(CS(C)(=O)=O)C(=O)N1CCC(Cn2cc(CN3CCOCC3)nn2)C1 75682,C1(CNC(CCC(C)SC)=O)CN(C(=O)Cc2ccnn2C)C2CCCCC12 75683,Nc1cc(C(=O)NCC23CC(NC(=O)C(O)CN4CCCC4)(CO2)C3)ccc1F 75684,C(=O)(CC(C)C(C)(C)C)N1CC(O)(CN(C(C(n2cnc(C#N)n2)CC)=O)C)C1 75685,CC1CN(C(c2ccc(Cl)[nH]2)=O)CCN1C(C1CC(CC(F)F)C1)=O 75686,C1(NC(=O)CN(CCO)CCO)CC2(C1)CN(C(c1ccc(Br)cn1)=O)C2 75687,c1(C(=O)NCC2N(C(c3cccc(C)c3C)=O)CC(O)C2)cc2c[nH]cnc-2n1 75688,Cc1cccc(CN(C(=O)CCCCNC(C2COCC2C(N)=O)=O)C)c1 75689,C(=O)(CC(O)CC(C)C)N1C(CC)C(NC(=O)CCCC(F)F)CC1 75690,c1(CNCc2nc(C(C)(C)C)sc2)cc(I)ccc1F 75691,C12(NC(C(CC)NC(C)=O)=O)CC(C1)N(C(=O)Cc1ccns1)C2 75692,C1(C(=O)NCC(C)NC(=O)OC)C=CC(NC(C2CCSC2)=O)C1 75693,C(c1ccc(O)cc1)=CC(=O)NCC(CN(C(=O)C(C)(C)n1cccn1)C)O 75694,N1(C(C2=CCCCC2C)=O)CCN(C(=O)CCc2cncnc2)C2(CCC2)C1 75695,Nc1nc(C(=O)NCCCCNC(=O)C2=NNC(C(F)(F)F)C2)ccc1[N+](=O)[O-] 75696,N1(C(CCCC(C)=O)=O)CC(NC(c2ccc(NC=O)cc2)=O)CC12CCOC2 75697,Cc1nnc2n1C(C(=O)NC1(CCNC(=O)Cc3ccc(F)c(F)c3)CC1)CC2 75698,N1(C(Cc2cccc(OC)c2)=O)CCCC(NC(C2CC(N(C)C)C2)=O)CC1 75699,Cc1ccc(NC(=O)CN(C(=O)CNC2CC(=O)N(C)C2=O)C)cc1C 75700,c1(OC)cc(=O)n(C)cc1C(=O)N(C1CN(C(C2OCC3CCCCC23)=O)C1)C 75701,C1(NC(=O)CC2CC(F)(F)C2)CC2CC1CN(C(c1cccc(CO)c1)=O)C2 75702,N1(C(CC2N(C)CCCC2)=O)CC2CCCC1C2CNC(=O)CCCC1CCC1 75703,N1(C(C(COC)C)=O)CCC(NC(c2ncc(F)c(OC)n2)=O)C(OCC)C1 75704,C1(CNC(=O)CC2CCCC2(F)F)CC2(CO1)CN(C(c1cccc(=O)o1)=O)C2 75705,C1(C(=O)NC(C2CN(C(=O)C(n3ccc(C4CC4)n3)C)C2)C)CCCC1(F)F 75706,c1(C(N2C3C(NC(C4CCCN4C4CC4)=O)CC(C3)C2)=O)ncn2ccccc12 75707,CCCC(C)(C)CC(=O)NC1CC2CCC1(NC(=O)Cc1ncc(CC)[nH]1)C2 75708,N1(C(c2nn(CC)c(C3CC3)c2)=O)CC(NC(c2ccnnc2)=O)CC2(CC2)C1 75709,N(C1CCc2ccccc21)C(CC(C)CNC(c1ncccc1Cl)=O)=O 75710,C1(C(=O)NC(CNC(c2cnc(C(C)OC)s2)=O)(C)C)CCc2n[nH]c(C)c2C1 75711,CS(=O)(=O)C1CC(CNC(=O)C(N)C2CSC2)C1 75712,c1(C(C)C)cccc(F)c1C(=O)NCCC(C)NC(c1cnc(Cl)[nH]1)=O 75713,C1(CCNC(C2C(C)(C)CC2)=O)(NC(C2CCC=CCC2)=O)CCOCC1 75714,c1(C(=O)NCC2C(NC(c3ccc(Cl)s3)=O)CCC2)coc2c1C(O)CCC2 75715,c1(N2CCC(C(N)=O)CC2)nc(N2CCN(c3ccncn3)CC2)c2c(n1)CCS2 75716,C(=O)(C(C)(C)CN1CCCC1=O)N1CCC(N(C)CC23CC(Cl)(CO2)C3)C1 75717,C1(NC(c2cnn(CCN(C)C)c2)=O)CCCN(C(C2(CF)CC2)=O)CC1 75718,C1(CC(=O)NCCC2N(C(CCC(=O)N(C)C)=O)CCCC2)CCCCC(=O)N1 75719,N1(C(C2CCCN(C)C2)=O)CCC2(C=C(C(=O)NC(c3cscn3)CO)C2)C1 75720,Cc1c(NC(=O)C(Cc2cocn2)NC(=O)OC(C)(C)C)cc(Br)cc1C(=O)O 75721,N1(C(CC2N(CC)CCC2)=O)CCN(C(C2(F)CCC2)=O)CC1c1nccn1C 75722,CC(CN=c1[nH]c2c(c(=NCCn3cc(Br)cn3)[nH]1)CCC2)c1ccc(Br)cc1 75723,c1(C(N2C(C)CCC(NS(CC)(=O)=O)C2)=O)ccc(Cl)c(OC)c1F 75724,c1(CCC(=O)NC(C)(CNC(=O)C=Cc2cn[nH]c2)CO)cccc(O)n1 75725,Cc1ccc(SC(C)C(=O)NCC2C3CN(C(c4ccc(CO)o4)=O)CC23)cc1 75726,C(=O)(CC1=NNC(=O)C1)N(CCCCCCNC(c1c(OC)cc(Cl)cc1)=O)C 75727,c1(C(=O)NCCCCCN(C(C(C(C)C)C)=O)C)ccnc2ncnn12 75728,Cc1cncc([N+](=O)[O-])c1N1CCC2(CC(NC(=O)COc3cnn(C)c3)C2)C1 75729,CC(C)C(O)CC(=O)NCC1CCN(CCOc2c(Cl)cccc2Cl)CC1 75730,C1(C2CC2)(CC)CCCN1C(=O)NC12CCC(C(CCC)CCC)C1C2 75731,c1(N(C2CC3CCC(C2)N3)CC2(S(C)(=O)=O)CCC2)ncnc2[nH]cnc12 75732,C(N(Cc1ccccn1)N1CCC(c2ccccc2)C1C)c1c(C)noc1C 75733,C1(NC(c2cnc(CC(C)C)[nH]2)=O)CCCC12CN(C(c1cc(Cl)ccn1)=O)C2 75734,C12(NC(C(C)S(N)(=O)=O)=O)CCCN(C(c3cnn(C4CC4)c3)=O)CC1C2 75735,C1(C(N2C3(CNC(C4(COC)CC=CC4)=O)CC(C2)C3)=O)CCCCCS1(=O)=O 75736,Cc1ccc(F)c(C(=O)NCC2(CNC(=O)CC3CC=CC3)CCC2)c1 75737,N1(c2c(OC)cncn2)C2CCC1CC(NC(=O)C=Cc1scnc1C)C2 75738,c1(C(=O)NC(CN(C(=O)CC(C)N2CCCC2=O)CC)C)nc2cnccc2s1 75739,c1(C(=O)NC(CC=C)CNC(=O)CCC#N)ccc(Cl)nc1OCC=C 75740,C1(C(N(CC=CC(N2CC(C(N)=O)C2)=O)CC)=O)CC(=O)C12CCC2 75741,C(=O)(C1SCCc2sccc21)N(CC(C)(C)CNC(=O)CCc1nccs1)C 75742,c1(C(N2CCN(C(C(CC)SC)=O)CC2)=O)ccc2nc[nH]c2c1 75743,N1(C(Cc2cccc(C)c2C)=O)CC2(CCC(CNC(=O)C(C)N3CCC3)O2)C1 75744,C=CCCCCC(=O)N1CC(CCNC(=O)CN2CCC(C)C2)C1 75745,C1(NC(C(N2CCN(C)CC2)C)=O)CCN(C(=O)CCCC2CC2)C1C1CC1 75746,c1(CN2C(C(N3CCCC3c3ccc(Cl)s3)=O)CCC2)ccc2ncsc2c1 75747,C(=O)(CC(C)C(=O)N(C1CN(C(=O)C(C)(C)c2ccnn2C)CC1(C)C)C)OC 75748,Cc1c(C(=O)NC2CCCC(NC(=O)C=CC(C)C)C2)nnn1C1CCOC1 75749,c1(N2CCC(CC)(CO)C2)ccc(Br)c(S(=O)(=O)NC(C)C(C)(C2CC2)OC)n1 75750,C1(C)(C(N2C(C3(NC(C4C(C=C)C4)=O)CC3)CCCC2)=O)CCN(C)C1=O 75751,N1(C(C(C(C)C)O)=O)CCN(C(C2CCC(O)CN2C)=O)C(CCO)C1 75752,c1(NC(C2C3CN(C(c4ccc(O)c(O)c4Cl)=O)CC23)=O)cc2cccnc2[nH]1 75753,C(N=c1[nH]c(N2CC=C(C)CC2)nc2c1CCCCC2)c1c(OC)c(Cl)ccc1 75754,C(C)(C)(CCN=c1[nH]c(N(C)Cc2nccn2C(F)F)nc2c1SCC2)OC 75755,C1(F)(C(=O)OC)CCC(CN(CCN(C(=O)CCc2ccncc2)C(C)C)C)C1 75756,N1(C(C2(C#C)CCCC2)=O)CCC2CCC(NC(=O)CS(=O)(=O)NC3CC3)C1C2 75757,C1(Cn2cc(C3CCCN(C(c4c(C)ccs4)=O)C3)nn2)CCCCC1(F)F 75758,N1(C(=O)NCC#C)CCC(N(CC(O)CC)C)C1 75759,c1(C(N2CC(O)(CNC(C(CSC)O)=O)C2)=O)ccc(Cl)cc1O 75760,C12(C(N3CC(C)N(C(c4c[nH]nc4S(N)(=O)=O)=O)CC3)=O)CCN(C1)S(=O)(=O)C2 75761,c1(C(=O)NC2CCCC(NC(=O)C3=CSCCO3)C2)c(F)cccc1[N+](=O)[O-] 75762,c1(CNC2C(C(=O)Nc3cc(CC)n[nH]3)CCCC2)ccc(OC)nc1Br 75763,C(=O)(C(F)CC(C)(C)C)NCc1nn(C)c(C(N2CCC(C)(CCO)C2)=O)c1 75764,N1(C(C(c2ccnn2C)NC(C(CC)O)=O)=O)CCCC(C2CC2)CC1 75765,C=C(C)CCCC(=O)NC(C)CC(C)NC(c1ccc(-c2cccs2)cn1)=O 75766,C(CC(C)(C)CNC(=O)CC1CCC(F)(F)C1)NC(Cc1c(C)ccs1)=O 75767,C1(C(=O)NC(C)(CNC(=O)C(C2CCCCC2)O)CO)CCCCS1(=O)=O 75768,Cn1ncc(CCC(=O)NCC2CC(CNC(c3cnn[nH]3)=O)CO2)n1 75769,N1(C(C2CC(OC)(OC)C2)=O)CC2COCC2(C(=O)NC2CC(F)(F)C2)C1 75770,c1(CCC)c(C(N2CCC(C)(CNC(=O)C(C)OC)C2)=O)nnn1CC 75771,C(=O)(C1=CC2CCC(C1)C2)N1CCCN(C(C(CCC)c2ccccc2)=O)C(C)C1 75772,c1(CCNC(CN(c2ccncc2C(F)(F)F)CC)=O)ccc(Br)cc1[N+](=O)[O-] 75773,C1(NC(Cn2cc(C(C)O)nn2)=O)CC(CNC(=O)Cn2ccnn2)C1(C)C 75774,C1(NC(C2CCCCO2)=O)CN(C(c2ccc(C(F)F)o2)=O)CC12CCC2 75775,CN1CCN(C(c2ccccc2C2(C)CC2)=O)C(CNC(c2c[nH]nc2Cl)=O)C1 75776,c1(NC(C(CO)NC(c2cnc(OC)nc2)=O)=O)ccc(C#N)cc1O 75777,S(=O)(=O)(c1nc(N2CCC=C(Br)C2)ccc1Br)N1CCC(COCC)C1 75778,c1(C(=O)NCC2CCC(NC(C(C)SCCCC)=O)C2)c(O)ccc(Cl)c1F 75779,c1(C(N2C3CN(C(C4C(OC)CC4)=O)CC2CC3)=O)c([N+](=O)[O-])c(C)nn1C 75780,c1(OC)nc(Cl)ccc1CNC(c1cc(N)ccn1)=O 75781,CC(C)CC(CNC(=O)Cc1ccsc1)NC(C12CC(CC(F)F)(C1)C2)=O 75782,C(CN=c1nc(OC)c2nc[nH]c2[nH]1)C1CN(C(C(CC)CC(F)(F)F)=O)C1 75783,c1(CCC(=O)NC(C(=O)N2CC(C(C)OC)C2)CO)cccnc1 75784,c1(C(N(CCC(C)NC(c2ccc(CCC)s2)=O)C)=O)ccn(C)c1C1CCC1 75785,C(=O)(C1=NN(C(C)C)C(=O)CC1)NC1CCN(C(C(CC#C)O)=O)C1CC 75786,C(=O)(C(C)(C)CNC(C1CCN(C(=O)COC2(C)CCC2)C1)=O)NC 75787,CCC(C)(CCC(C)C)C(=O)N1CC(O)CC1C(=O)NCc1cccc(Cl)n1 75788,N1(C(C2(C(C)=O)CC2)=O)CC(CNC(=O)Cn2cnc([N+](=O)[O-])c2)OC(C)(C)C1 75789,C(=O)(CCC(C)C)NCCn1c(SC(c2ccccc2)C(=O)OCC)nnc1 75790,c1(C(N2CCN(C(CCOC)=O)CC2CC#N)=O)cccc([N+](=O)[O-])c1OC 75791,C1(CC=C)(C(=O)NCC2(CCC)CCC2)CCCN1C(=O)C(C)CC#N 75792,c1(C(=O)NC(c2ccccc2Cl)C)nc2ccccn2c1-c1ccoc1 75793,Cc1cc(C(=O)NC2C3CC(NC(=O)C(O)c4ccsc4)CC23)nc(C)c1 75794,CC1Cc2ccc(F)cc2C1Nc1cc(I)ccc1F 75795,C1(NC(C(Cn2cncn2)OC)=O)CCOC(CNC(c2cc(Cl)no2)=O)C1 75796,N1(C(C2C(c3onc(C(C)C)n3)C2)=O)CCC(F)C(F)C1 75797,N1(C(CCSC)=O)CC(CNC(c2sccc2-n2cnnn2)=O)CCC1C 75798,C1(C(=O)Nc2cc(O)n[nH]2)CN(Cc2cccc(Br)c2Cl)CCC1O 75799,c1(C(N2CC(NC(C3ON=C(CC)C3)=O)C(C)C2)=O)cccc2c1CCC(=O)N2 75800,S(=O)(=O)(c1cnc(NCCCOc2cncc(Cl)c2)cc1C)NCCC(=O)NC 75801,N1(C(=O)Cn2cncn2)CC2CCN(C(=O)C3=CS(=O)CCC3)C2C1 75802,C(=O)(C(C(C)C)C(C)C)N1C(CCNC(c2ccc(CC)nc2)=O)CSCC1 75803,c1(CC(N2CCN(C(CC3(C=C)CC3)=O)CC2CO)=O)ncn2c1COCC2 75804,c1(C(C(C)C)OCC)noc(CS(=O)(=O)Cc2sccc2Cl)n1 75805,C1(O)(C(C)NC(Cc2cnc(C)s2)=O)CCN(C(c2ccc(Cl)s2)=O)C1 75806,N1(C(N(C)C)=O)CCCC(C(=O)NC2CCC(NC(=O)Cc3cn[nH]c3)C2)C1 75807,N1(C(N(c2ccc(C)cc2Br)C)=O)CC2(CCCC2)C1C(C)C 75808,C1(C(=O)NCC2CN(C(=O)CN3CCC(CF)C3)C2)CC2CCC(C1)C2(F)F 75809,Cc1ccc(C(N2CCCC(C(=O)NC3(C)CC(C(=O)O)C3)C2)=O)c(Cl)n1 75810,C(=O)(C(C)(O)CC)N(CC(CNC(C(CC)NC(N)=O)=O)(C)C)C 75811,C(=O)(C(C)(C)CC(C)(C)C)NCc1scc(C)c1.N12CCC(C1)C2=O 75812,c1(C(N2CCC3(NC(c4cc(C)cc(F)c4)=O)C(C2)C3)=O)ccc2nc[nH]c2c1 75813,c1(C(CCN(C)NC(=O)C(=O)NCC(F)(F)F)NCC(=O)NC2CC2)ccccc1 75814,Cn1cnc2c(C(N3CCC(CNC(C4CCC5CC45)=O)CC3)=O)[nH]nc2c1=O 75815,N1(C(C2C(C)C2)=O)CCCC(CNC(=O)CS(=O)(=O)Cc2ccccn2)CC1 75816,Cc1cnc(C2CCCN2C(CCC2(C)CC2)C(=O)NC2CCCCC2)c(C)c1 75817,C1(C(=O)NCC2CCCC(OC)C2)N(C(c2n[nH]cc2C)=O)CCC1(C)C 75818,c1(C(=O)NC(CC)CNC(c2cc(C(F)F)[nH]n2)=O)cnccc1C1OCCO1 75819,Cc1ccn(CC(=O)N(CCCCNC(=O)CSC(C)C)C)n1 75820,N1(C(=O)Cc2ccoc2)CC2CC1CCN2C(=O)C(O)Cc1ccccn1 75821,c1(OCC)ncccc1C(=O)Nc1cccc(NC(C2CC(O)C(F)C2)=O)c1 75822,Cc1ccsc1C(=O)NCCCCN(C(=O)C(c1cccnc1)N(C)C)C 75823,c1(C(=O)NC(C(C)NC(c2cc(C(C)=O)c(C)o2)=O)C)c(C)nc(C)nc1C 75824,Fc1ccc2c(c1)CCC2N=c1[nH]c(=NCc2ccnnc2)c2ncccc2[nH]1 75825,Cc1ccc(C(=O)NC2CN(C(C3(CCF)CCC3)=O)CC23CC3)cc1O 75826,c1(C(N2C(CNC(C(C)(C)OC)=O)CCC2)=O)cccnc1I 75827,C1(NC(=O)C=Cc2cscn2)C2CC3C(C2)C13C(=O)NC1CC(=O)N(O)C1 75828,c1(N(c2n(CC=C)c(-c3scnc3C)nn2)C)ccc(OCCCC)c(Cl)c1 75829,N1(C(C=CC)=O)CCN(C(=O)C=CC2CCC2)C2CCCCC12 75830,N1(C(C2C(C)C2)=O)CC2CC1C2CN(C(c1ccccn1)=O)Cc1ccccc1 75831,C1(C(=O)NC2CCN(C(Cc3n(C)ccn3)=O)C2)CCc2ccccc2C1O 75832,C1(NC(c2n(CC)ccn2)=O)COC2(CNC(C3(C(C)C)COC3)=O)CC1C2 75833,C1(CN(C(=O)CC2CCCSC2)C)CCN(C(c2nnsc2N)=O)CC1 75834,C1(C(=O)NCC(C(C)(C)C)OC)CCCCCCN1C(=O)C=C(C)c1ccco1 75835,c1(OC)cc(Cl)c(NC(=O)C(N2CCC(C(=O)NC(=O)C3CC3)C2)=O)cc1C 75836,c1(CC(=O)N(CC(C)(C)NC(=O)CC2CC2(Cl)Cl)C)ccccc1OC(F)F 75837,Cc1ccc(CNc2csc(-c3cc(C)[nH]n3)n2)cc1 75838,c1(CC)ccccc1CC(=O)NCC1(NC(C2CCCCC2O)=O)CC1 75839,N1(C(c2ccc(C)cc2O)=O)CC(F)(F)CC1(C)CNC(=O)C(C)C(C)(C)C 75840,Cc1ccccc1CC(=O)NCC(O)CNC(=O)C=Cc1csc(Br)c1 75841,S(=O)(=O)(c1cncc(Br)c1)NC(C1C(C(N2CCN(CCC(C)C)CC2)=O)C1)=O 75842,c1(CC)cc(C(N2CC(C(F)Cn3cc(-c4ccc(Cl)s4)nn3)C2)=O)n[nH]1 75843,c1(NC2CN(C(c3cc(C)sc3C)=O)CC2C)ncnc2c1nnn2C1CC1 75844,c1(C(=O)NC(CCOC)CNC(=O)C=C(Cl)Cl)cn(C)c(=O)c2ccccc12 75845,C1(CC(=O)N(CCN(C(=O)CC(C)n2cccc2)CC)CC)CCCC(F)(F)C1 75846,Cc1c(C(N2CC(C3(NC(=O)CSCCN(C)C)CC3)C2)=O)cncc1Cl 75847,N1(C(CCSCC)=O)CCC2OCCN(C(c3cc(C)cc(O)c3)=O)C2C1 75848,Cc1ccc2cccc(C(=O)Nc3ccnc4ncnn34)c2n1 75849,N1(C(CCCCNC(N)=O)=O)CC(C2CCCN(C(c3ccc(F)cn3)=O)C2)C1 75850,c1(C2C(F)(C(=O)NCCNC(c3coc(Cl)n3)=O)C2)ccccc1F 75851,Cc1nc(C)n(CCC(N2CCC(N(CCO)C(C3CC(C)(C)O3)=O)C2)=O)n1 75852,C1(C(=O)OC)CCCN(C(c2ncc(OC)cn2)C(=O)NCC2CCOC2)C1C 75853,C1(OCC(N2CCC(C(N3CC(OC)C3)=O)(OC)C2)=O)CN2CCC1CC2 75854,C1(C(=O)NCCC(c2ccncc2)(C)C)(OCC)CCN(C(=O)OC(C)(C)C)C1 75855,C1(C(N2CC(C(C)C)OCC2)=O)CC(C)CN(C(=O)C(C)(C)CC#N)C1 75856,c1(C(=O)NCCCCN(C)C(C2CC(N(C)C)C2)=O)[nH]nnc1-c1ccnn1C 75857,N1(C(C2(SC)CCC2)=O)CCCN(C(C2CCN2S(C)(=O)=O)=O)C(C(C)C)C1 75858,N1(CCNC(C=CCN(C)C(c2cnc(Cl)s2)=O)=O)CCCOC1=O 75859,C#CCC(CC(=O)NCC1(CCO)CCCC1)NC(C1(C)C=CCCC1)=O 75860,Cc1n[nH]c(=NCC2CC(C)N(C(c3cc(O)nn3C)=O)C2)s1 75861,S(=O)(=O)(c1cc(C(C)C)cc(Br)c1)Nc1ncc(-c2ccc(C)cc2)s1 75862,Cc1cc(Br)c(F)cc1CN1CC2C(C1)N2C(=O)C(C)(C)CCl 75863,C1(CC)CN(C(=O)CC2CC3(CC3)CO2)CCC1NC(=O)CS(=O)(=O)NC 75864,c1(C(=O)NCCCC(C)NC(C2(O)CC2)=O)ccc(CNC(N)=O)cc1 75865,Cc1ccc(C(c2nnnn2Cc2ccccc2)NCC(F)CO)cc1Br 75866,c1(C(=O)NCC2(COC)CN(C(C3CC3C3CCCO3)=O)C2)cc(C(F)F)[nH]n1 75867,n1(CC(C)NC(C(c2ccccc2)OC)=O)cc(CN(C)C(C)=O)nn1 75868,CC1CCCC(N(C)C(c2ccc(CNC(=O)CCCC3CCC3)s2)=O)C1 75869,N1(C(CS(C)=O)=O)CC2CCC1CN2C(=O)CCc1cc(F)c(F)c(F)c1 75870,N1(C(C(C)=CC2CC2)=O)CC(CNC(c2c(C)ncnc2C)=O)CC(C)(C)C1 75871,Cc1cnc(-n2nc(CCCOc3cc(F)cc(F)c3)nc2CC(F)F)cc1Cl 75872,C=CC(C)(C)C(=O)NCCN(CC(C)O)C(C1CC1C)=O 75873,c1(C(N(C(CCNC(c2nn(CC)c(=O)cc2)=O)C)C)=O)cc[nH]c2nccc1-2 75874,C1(NC(CCC2C(C)(C)C2)=O)CCC(NC(=O)C(O)C2CCCC2)CC1 75875,C1(C(=O)NCC2N(C(C(C)OC3CCCC3)=O)CC2)CCCN1C 75876,c1(C(N2CCC(NC(C(F)=CCC)=O)C(F)C2)=O)c(C)cc(Br)cc1C 75877,c1(C(N(CCC)CCNC(C2(C)CCCC2)=O)=O)ccc(CCN(C)C)cc1 75878,Cc1cccc(C(=O)NC(C)C=CC(N2CCN(C)C(=O)C2)=O)c1C#N 75879,N1(C(C(C(C)C)SCC)=O)CC(C)(C(=O)N(CC(=O)NC)C(C)C)CC1(C)C 75880,C1(C)(C(=O)NC2C(OC)CN(C(c3cc(C4CCC4)on3)=O)C2)CCCNC1=O 75881,N1(C(C2CC(F)C2)=O)CCN(C(C2CC(O)(c3ccccn3)C2)=O)CC1CO 75882,C(=O)(CC(CNC(=O)CC1(C)CCOCC1)C1CCC1)OC.Cc1cscc1CN 75883,CC1(NC(c2c[nH]cc2Br)=O)CCN(C(=O)CSc2n[nH]c(O)n2)CC1 75884,S1(=O)(=O)c2ccc(cc2)N1.N1(C(C)CO)CC2(CCC2)C1C(=O)NC1CC1 75885,C(C(C(C)C(C)C)NC(c1cccnc1C(F)(F)F)=O)NC(CNC(C)=O)=O 75886,c1(C(=O)NCc2cccc(NC(C3(C)C(C)OCC3)=O)c2)ccc(CO)c(Cl)c1 75887,Cc1cc(C(=O)N(CCCCN(C(=O)CCOc2ccc(F)cc2)C)C)c(C)[nH]1 75888,CC(C)(CCCN=c1nc(CC2CC2)[nH]s1)NC(=O)C(C1CCOCC1)O 75889,N1(C(CCC=CCC=C)=O)CCCN(C(=O)CC2(n3cccn3)CC2)C(C)C1 75890,C1(C(=O)NC(C=C)C)CN(C(=O)CC(C)CCC)CC12CC2 75891,c1(SC)cc(C(=O)NCC(C)CNC(c2ccc(C(C)C)o2)=O)ccc1F 75892,c1(C(c2nnnn2C)NCc2cnc(C)s2)ccc(Cl)c(C(F)(F)F)c1 75893,Cc1n[nH]c(=NCC2CCN(C(=O)CCCOc3cccnc3)CC2C)o1 75894,C1(C(=O)NCc2c(C(=O)NCC3CCC=CO3)occ2)CC2(CCC2O)C1 75895,c1(C(=O)NCC(CC)NC(=O)CC2CCn3cncc3C2)cc(Cl)c(O)cc1C 75896,C1(O)(CCNC(CC2C(C)C2)=O)CCN(C(c2ccc(N)cn2)=O)CC1 75897,c1(C(N2C(CN(C(CC(=C=C)C)=O)C)CCCC2)=O)ccc2c(c1)CCO2 75898,C=C(Cl)C(C)(C)C(=O)N1CCCCC(NC(=O)C(C(C)C)NC(=O)COC)C1 75899,Cc1csc(C(=O)NCCn2ccc(C(=O)N(CC3=CCSC3)C)c2)c1 75900,N1(C(c2c(C)nn[nH]2)=O)CC(NC(C2CCCN2c2nccs2)=O)C2CC2C1 75901,c1(C(N(CC(CNC(c2nn(CC)c(C)c2)=O)C)C)=O)[nH]cc2c1CCS2(=O)=O 75902,c1(C(N2CCC(CN(C)C(c3ccn(CC#N)n3)=O)C2)=O)cc2cnn(C)c2s1 75903,C1(C(=O)NC(C2(O)CN(C(C34CC5CC3C4C5)=O)C2)C)CCC(C)(C)C1 75904,C1(NC(c2c(CC)nc[nH]2)=O)CC2CC1N(C(=O)CC(O)c1cnc(Cl)s1)C2 75905,c1(C(N(CC(C)NC(c2c(Cl)ccc(C)c2)=O)C)=O)cccc2cnnc(O)c12 75906,c1(C(=O)NC(CNC(c2c(C)nn(C3CC3)c2)=O)CO)c(C)oc(C)c1C 75907,c1(C(=O)NCC(C)(C2CC2)NC(c2cc(CO)[nH]n2)=O)cc2n(n1)CCO2 75908,C(c1c(C)noc1C)=CC(=O)NC(CC)(C)CCNC(=O)C(C)=C(C)C 75909,c1(C(N2C3C(NC(CC=C=C)=O)C(C3)C2C)=O)cc(C)c(F)cc1F 75910,C1(CC(=O)NCCSC)CN(C(C2CC3C=CC2CC3)=O)C(C)(C)C1 75911,c1(CNC(=O)COC(F)F)cnn2c1CN(C(=O)CC1C=CCCC1)CC2 75912,c1(C(N2CC(F)CC(NC(CSCC=C)=O)C2)=O)ccnc(S(N)(=O)=O)c1 75913,C(=O)(C(O)C1=CCCCC1)NCC1(F)CN(C(c2ccc(NC)c(F)c2)=O)C1 75914,c1(CN2C(C(=O)NCc3ccn(CC)n3)CCC2)c(F)cc(I)cc1F 75915,N1(C(c2oc(CC)c(C)c2)=O)CCC2(CC1)CC2CNC(c1csnc1OC)=O 75916,N1(C(c2c(C)cc(C3CC3)nc2)=O)C2CCC1CN(C(C1CCCC(C)C1)=O)C2 75917,c1(NC(C(C(C)C)CNC(C2CCC(=O)NC2)=O)=O)ccc2c(c1)COC2 75918,C1(C(N(CCCNC(C2(NC(N)=O)CC2)=O)C)=O)CCCCC1c1nncn1C 75919,C1(C(N(C2CCC2)CC)=O)CC(C)N1C(=O)CCc1cncnc1 75920,C1(CCNC(Cn2c(C)ccn2)=O)CC(F)(F)CN1C(c1c[nH]cc1Br)=O 75921,C(c1cccc(F)c1F)=CC(N1CCC(O)(CNC(C(C)(F)F)=O)C1)=O 75922,C(=O)(CCCCC(C)C)NCC(C)(C1CC1)NC(COc1cccc(CC)c1)=O 75923,c1(OC)cccc(C2CCN(C(C3CCCSC3)C(=O)NC3COC3)C2)c1 75924,c1(C(=O)NC(CC=C)CNC(c2cc(C)[nH]n2)=O)cc(C)c2ncccc2c1C 75925,CC12CCC(C(=O)NC3CN(C(c4ncoc4C4CCCC45CC5)=O)C3)(CC1)C2 75926,C(CCC(C)C)(C(=O)NC1CC2CC2C1)NC(C(C(CC)C)=O)=O 75927,CC1CC(NC(c2cnoc2)=O)CCN1C(c1cnns1)=O 75928,CC(CNC(C1C(C)C1C)=O)C(=O)NC(C)C(C)F 75929,CCC(CC(=O)Nc1ccc(N(C(=O)C(=O)NC)C)cc1)C1CCC1 75930,N1(C(CC=CCC)=O)CC(NC(=O)C(C(C)C)N2CCCC2=O)C2(CC2)C1 75931,c1(C(N2CC3(C)CC2(C(=O)NCCC2CCSC2)C3)=O)ccc2n[nH]cc2c1 75932,C(=O)(CC1=CCCC1)N1C(C)CC(NC(=O)C(c2ccc(Cl)cn2)(F)F)C1 75933,c1(C(=O)NCC2N(C(c3c(C)nc(C)[nH]3)=O)CCCC2)cc(Cl)c(F)cc1F 75934,CC1(C)CC(CNC(c2cn3cnnc3cn2)=O)CN(C(=O)COC(C)(C)C)C1 75935,c1(C(=O)NCC(CCCC)NC(=O)CC2CSCCS2)cccc2scnc12 75936,c1(C(N2CC(CC(=O)Nc3nccc(Br)c3Cl)OCC2)=O)cc(F)c(F)cc1O 75937,N1(C(C(C)=C2CCC2)=O)CC(O)CC1C(=O)NCC(c1ccccc1)C1CC1 75938,CC1CC(CNC(c2c(Cl)cnn2C)=O)CCN1C(c1cnsc1)=O 75939,CCC(C)C(O)C(C)C(=O)Nc1cccc(NC(C2(OC(C)=O)CCCC2)=O)c1 75940,c1(C(N(CCNC(C2CC(=O)N(C)C2)=O)CC)=O)cnc2c(C)cccn2c1=O 75941,N1(C(C2CCC(C(N)=O)C2)=O)CCCC(NC(C2CN(CC(F)(F)F)C2)=O)C1 75942,C12(C(=O)NCCCCC(C)NC(C3CSCC(=O)N3)=O)CCC(C1)C2(C)C 75943,c1(C(N2C(CCNC(c3ccc(C)o3)=O)CSCC2)=O)ccc2c(c1)OCO2 75944,C1(C(=O)NCCOCCOCCNC(C2C(C)C2)=O)COc2ccccc2O1 75945,N1(C(c2cncc(Br)c2)C(=O)NCC=C)CC(C)(C)c2ccccc21 75946,CC1C(NC(C2CC3(CC3)C2)=O)CCCC1n1cc(C2CC=CCC2)nn1 75947,N1(C(C(CC(=C)Cl)NC(=O)CCC2CCC2)=O)CCNC(=O)CC1C 75948,c1(C(N2CC=CC(NC(c3c(C)onc3Br)=O)C2)=O)ccc(Cl)c(N)c1 75949,c1(C(N2CC(C(C)(F)F)OCC2)=O)c(F)cccc1I 75950,CC1COCCN1C(C1CCCN1C(=O)Cc1ccccc1Cl)=O 75951,CC1=CCSC1C(=O)NCCC1CCCN1C(=O)CC1CNC(=O)O1 75952,C#Cc1ccnc(C(=O)NC2CC(CCNC(c3ccc(C(F)F)s3)=O)C2)c1 75953,C1(N(C(C#CC(C)C)=O)C)CC2CC1N(C(=O)C(n1cc(Cl)cn1)C)C2 75954,c1(-n2cc(CC(N3CCOCC3C3CCCC3)=O)nn2)ccc(C(=O)O)cc1F 75955,c1(OC)cc(C(=O)NCC2(O)CC(CNC(C3(OC)CCSC3)=O)C2)cc(Cl)c1 75956,Cc1cc(Cl)c(C(=O)N(CC(O)CN(C)C(c2cnc(O)c(F)c2)=O)C)cc1F 75957,C12(C(N3CC(NC(C4CN(C(=O)OCC)C4)=O)C3)=O)CCOC1CC(=O)NC2 75958,c1(C(C(=O)NCC(C)NC(=O)C=Cc2ccoc2)O)ccc(Cl)c(Br)c1 75959,C=CCCCCCN(C)C(=O)NC1(c2ccccc2)CCCCO1 75960,c1(C(=O)NCC2N(C(CN(C)CC)=O)CCN(C)C2)cc(Cl)c2c(c1)OCCO2 75961,c1(C(N2C(CNC(c3nncc(C)c3)=O)CCC2)=O)ccc2c(c1)nc(O)n2C 75962,c1(CNC(=O)CN2CCOCC2)ccccc1CNC(c1cc(Cl)c[nH]1)=O 75963,N1(C(CN(CC)CC)=O)CCCCC1C1CCCN1c1ncnc2c1cnn2C 75964,C(=O)(CC1=CCCCC1)NC1CC(CCNC(C(C)(F)c2ccon2)=O)C1 75965,CCCCC(CNC(=O)OC(C)(C)C)NC(=O)CCN1CCNC(=O)C1 75966,CC1CCc2[nH]c(=NCC(C)(C)CC(F)(F)F)[nH]c(=NC3COCC3N(C)C)c2C1 75967,C(CC(=O)N(C)CCNC(C12COCC1C2)=O)(C1=CCCC1)OCC 75968,N1(C(c2cc(C)[nH]n2)=O)CCC2(CC1)CC2NC(=O)C(C1CC(F)(F)C1)O 75969,Cn1cc(C(=O)NCC2(NC(=O)CC3CCC(C#N)C3)CCC2)c2ccccc12 75970,C1(C(=O)NCCN(C(c2cnc(C)cc2Cl)=O)CC)CCC2(CCOCC2)O1 75971,N1(C(C(C2CCOCC2)C)=O)CCC(C(F)CNC(C2(C)CS(=O)(=O)C2)=O)CC1 75972,c1(CC(N2CCN(C(C(C)OC3CCOCC3)=O)CC2)=O)c[nH]c2ccccc12 75973,N1(C(CC(CCC)(C)O)=O)CCC2CCC(C1)N2C(C1(C)CCOC(C)C1)=O 75974,C#Cc1ccc(C(N2CCCC(CCNC(C3(CCO)CC3)=O)CC2)=O)nc1 75975,c1(COC)ncc(C(=O)NC2(C)CC(NC(=O)C(C)(C)c3ccno3)C2)c(=N)[nH]1 75976,c1(C(=O)NC(CNC(C(CC=C)CC)=O)C)cnc2cc(O)ccc2c1 75977,C(=O)(CCCC1CCNCC1)OCC(=O)NCC(C)C 75978,C1(NC(c2cnc[nH]2)=O)CC2CN(C(=O)CCc3ncc[nH]3)CCN2C1=O 75979,N1(C(CCCC(C)C)=O)CCCC2C(CCCN2C(c2ccnn2CCF)=O)C1 75980,C(=O)(CCC(C)N(C)C)N(C1CC(NC(CCC=C)=O)C1)C 75981,c1(C(=O)NC2(C)CN(C(C3C(C)CC3)=O)C2)cc([N+](=O)[O-])ncc1Br 75982,N1(C(CC(C)n2cccc2)=O)CCC2CN(C(C3CC4(C3)CC(O)C4)=O)CC2C1 75983,Cn1ncc(NC(C2CCC(CC(=O)NCc3csc(Br)n3)CC2)=O)c1C(N)=O 75984,C(=O)(C#CCNC(c1sccc1CC)=O)NCC=C 75985,C1(CC(=O)N(C)CC2CCC(NC(c3cncs3)=O)CC2)CC2(CCC2)CO1 75986,N1(C(CCc2c(C)cccc2)=O)CC2CC1CCN2C(c1cnn(C2CC2)c1)=O 75987,CCCS(=O)(=O)CC(=O)NCCCN(C(C1(C2CCCO2)CCCC1)=O)C1CC1 75988,c1(C(=O)NCC2CCN(C(=O)CSC(F)(F)F)C2)c[nH]c2cccnc12 75989,Cc1cc(OC(F)F)ccc1NC(=O)NC1CCN(CC(F)(F)F)C1 75990,c1(OC)noc(C)c1C(=O)NCCCC(C)NC(C12CCCCC1C2)=O 75991,N1(C(CS(=O)(=O)NC)=O)CCC(C)(C)C(NC(C2CNC(=O)C(C)(C)C2)=O)C1 75992,C(=O)(C#CC(C)C)NCCOCC(=O)NC(CC)C(N)=O 75993,C(=O)(N=c1cc[nH]c(CCO)c1)C1(O)CCN(C(=O)C=Cc2cnc[nH]2)C1 75994,C#Cc1ccc(OCC(=O)NC(C(=O)NOCC(C)(C)C)C2CCCO2)cc1 75995,C#CCC(CC(F)F)C(=O)NCC(C)(C)OCC(=O)NCC1(c2ccsc2)CC1 75996,c1(CSC)cc(C(=O)NC(C)CC2CN(C(=O)CCC3CCCCO3)C2)sc1C 75997,C12(C(N3C(C(=O)Nc4csc(Cl)c4)CCCC3)=O)CCC(CC1)CC2 75998,C1(NC(=O)C=CC2CCCC2)CCCCC1NC(C1C(F)(F)C12CC2)=O 75999,N#CC1(C(N2CCCC(NC(c3cccc4c3CCC4)=O)C2)=O)CC2(CCC2)C1 76000,c1(CC)cc(CC)[nH]c(=NCC(O)CNC(c2cn3c(n2)CCCC3)=O)n1 76001,C1(OC)CCN(C(=O)CC(C(C)C)NC(C2CCCN2C2CC2)=O)CC1(C)C 76002,c1(CC(N2C(C)CC(NC(=O)Cc3cnc[nH]3)C2)=O)c[nH]c2ccc(F)cc12 76003,c1(C(=O)NCC2CN(C(C3COC(=O)O3)=O)C2)ccncc1Br 76004,Cn1cc(C(=O)NCC2(NC(C3CC4C=CC3C4)=O)CCC2)c(C2CCCO2)n1 76005,C12(CNC(COCC)=O)CN(C(c3cncc(C)c3)=O)CC1(C(F)(F)F)C2 76006,N1(C(C2ON=C(C)C2)=O)CCN(C(c2ncn3ccccc23)=O)C2(CCC2)C1 76007,c1(C(=O)NCC(CN(C)C(C2CCSCC2)=O)O)ccc2c(O)nnc(O)c2c1 76008,Cc1nccnc1C(=O)NC(CNC(=O)CC1CC(n2cnnc2)C1)C1CCC1 76009,C12(C(N3CCCC(NC(=O)C=C4CCCC4)CC3)=O)CCCCC1C2(F)F 76010,CC(C)(C)CC(F)C(=O)NCC(=O)NCC(N1C(C)CC1(C)C)=O 76011,C=Cn1nccc1C(N1CC(F)CC1CNC(c1ccccc1)=O)=O 76012,C(=O)(CCCS(=O)(=O)N1CCCC1)N1CC(NC(c2cc(O)ncn2)C)C2C1C2 76013,CCC(C)(C)CC(=O)NCC1CC(NC(=O)C(c2ccccc2Cl)(C)O)C(O)C1 76014,C(C(COC)C(C)C)NC(c1c(C(C)NC(CN(CCOC)C)=O)noc1)=O 76015,n1(CC(=O)NC23CCC(C2)N(C(C2(S(N)(=O)=O)CC2)=O)C3)nc(C)ccc1=O 76016,c1(C(N2CC(NC(CCC#CC)=O)CC2(C)CC)=O)c[nH]c2c(C)cccc12 76017,N1(CC)CC2CCC1C2.c12ncc(o1)C(=O)N(C)CCC(=O)NC2C 76018,CCCCC(O)C(C)C(=O)NC(CCC(=O)NCCn1cc(CC)cn1)C(C)C 76019,c1(C(=O)NCCC2(C)CCN(C(C(CN(C)C)(F)F)=O)C2)ccnc2[nH]ncc12 76020,C(CN=c1[nH]c2c(c(=NCCOc3ccccc3)[nH]1)CSC2)C1(C)CCCO1 76021,N1(C(CC(CNC(=O)C(C)(C)C2(O)CCC2)OC)=O)CC2(CCC2O)C1 76022,C1(NC(C(CC)CC(C)C)=O)CCCCC12CCN(C(=O)CSC(F)(F)F)C2 76023,Cc1cc(O)ccc1C(=O)NC1CC(NC(=O)CSc2ccncc2)CC1O 76024,Cc1c(CC(=O)NCC(C)NC(C2CCCN2C)=O)ccc(Cl)c1Cl 76025,C(=O)(C1=CCCCC1P(C)(C)=O)N(C(CNC(c1cc(OC)c(C)cc1)=O)C)C 76026,C(=O)(C(CCC1CCCOC1)N1CCOC(c2cnn[nH]2)C1)NCCCC1(C)N=N1 76027,c1(C(=O)NC2CN(C(C3CC3(Cl)Cl)=O)CC2C(F)F)cnc(O)c2ncccc12 76028,c1(C(=O)NCC(CC=C)NC(=O)CCCCOC)cc(O)cc(F)c1F 76029,N1(C(c2cnc(C3C(C)C3)s2)=O)CC2(C1)CN(C(C13COC(CF)(C1)C3)=O)C2 76030,N1(C(c2ccc(SC)o2)=O)CCC(F)(C(=O)NCC2(O)CSC2)CC1 76031,c1(CC(C)=CC(=O)NCCOCC(N2CCOCC2)=O)ccc(C)c(C)c1 76032,[N-]=[N+]=NCCCC(=O)NCC1(CO)CCN(C(C2Cc3nncn3C2)=O)CC1 76033,C1(CC(=O)NCC(C)N(C(=O)CCc2ccccc2F)C)CCOC1(C)C 76034,C(CNC(=O)C1=CSCS1)(C(C)(C)C)NC(C(C)OCC)=O 76035,N1(C(C(CO)NC(N)=O)=O)CC2(CCCN(C(c3cc(C4CCC4)on3)=O)C2)C1 76036,C#Cc1ccc(OCC(N2CC(NC(c3cnc(C)cc3C)=O)CC2C)=O)cc1 76037,c1(C(N2CCC(N(C(c3nc(C)nn3C)=O)C)C(C)C2)=O)cccn2ccnc12 76038,c1(C(=O)NC2CCC(CNC(c3c(C)oc(Cl)n3)=O)C2)cc(O)cc([N+](=O)[O-])c1 76039,c1(CC)cc([N+](=O)[O-])c(C(=O)NC(CNC(=O)C(CC)OC)CO)cc1CC 76040,C(CCCCCC(=O)NCC(C)N(C)C(c1ccc(C(F)(F)F)c(F)c1)=O)SC 76041,N(C(=NCC1CCCN1CCCC)NCC(C1(O)CCOCC1)(F)F)C(C=C)C 76042,c1(NC(C2CCC(C(CC)(C)C)CC2)=O)cc(C)cc(Br)c1C 76043,C1(C(=O)NC2CCN(CCNC(C(C)c3cc[nH]n3)=O)CC2)CC2CCCCC12 76044,c1(N2CCC(=C)C2)ccn2ncc(S(=O)(=O)NC3CCC4CC34)c2n1 76045,c1(N(CC(N)=O)CC2(C)CCN2)ccc2ccccc2c1 76046,c1(C(=O)NCCC(C)NC(c2c(C)noc2C)=O)ccc2nc(O)[nH]c2c1 76047,C1(CNC(C(C)NC(C)=O)=O)CCN(C(=O)Cc2ccccc2Br)CC1 76048,C12(C(=O)NCC3C(C)CN(C(=O)Cc4cnn(C(F)F)c4)C3)CCOC(C)(C1)C2 76049,c1(C(N2CCN(C(=O)NC3CCCC(C(N)=O)C3)CC2)=O)c(F)cc(F)cc1Br 76050,C1(C(=O)NCCCCC(C)NC(=O)C=CC2CCC2)CCc2ccccc2N1 76051,c1(C(N2CCC(n3cccn3)CC2)C(=O)NC)ccc(S(C)(=O)=O)s1 76052,c1(OC)nsc(C(=O)NC2(CNC(c3nnn(C)n3)=O)CCCC2)c1Br 76053,C#Cc1cc(C(=O)NC2CS(=O)(=O)CC2NC(=O)C(C)CC(F)(F)F)ccc1C 76054,c12nc3n(c1Cl)CCN(C3)OC2.C(C(C(=O)OC)NC(=O)OC(C)(C)C)SCC 76055,c1(OC)cccc2c(CCNC(C3(c4ccc(F)cc4)CC(C)(C)C3)=O)c[nH]c12 76056,N1(C(c2ccc(CC)c(C(F)(F)F)c2)=O)CCCC2C1CCN2C(=O)C(C)OC 76057,C(=O)(C(C)CS(C)=O)NCC1(CNC(c2c(C)n[nH]c2C)=O)CC1 76058,C(=O)(C(C)(C)CC)NCC1(NC(c2cn(CCC3CC3)nn2)=O)CC(OC)C1 76059,C1(C(=O)NCC(CC(C)C)(C)C)CCN(C(=O)CCC(C)(C)F)O1 76060,CCC(O)C(C)(C)C(=O)NCC1(CN(C)C(c2cc(O)nc(Cl)c2)=O)CC1 76061,C=Cc1cncc(C(=O)NC(CNC(c2cnsn2)=O)CCCC)c1 76062,CC(C)C(O)C(=O)N1CCC(C(C)(O)CNC(=O)C(F)=C2CCCC2)CC1 76063,C1(C(=O)NCCOC(CNC(c2c(CC)n(C)nc2)=O)(C)C)CC2CCC(C1)C2 76064,C(CC(CNC(=O)CN1CCCCC1)NC(=O)C=C1CC(CF)C1)OC 76065,CC(C)(CC(F)(F)F)C(=O)N1CCCC(NC(C2Cc3nncn3C2)=O)CC1 76066,N1(C(c2cc(C(C)=O)oc2C)=O)CCCN(C(c2csnc2Br)=O)CCC1 76067,C1(C(=O)NCC(=C)C)CC(N(C(=O)CCC2CCC2)C)C1 76068,N1(C(C2CC2c2cccc(F)c2)=O)CC2CC1CN2C(C12CCC(CC1)C2)=O 76069,N1(C(CCc2cn(C)nc2)=O)CCCCCC1C(N1CC(CC2CC2)C1)=O 76070,c1(C(=O)OC)c(C)[nH]c(C)c1C(=O)C(C)ON(C(C)CO)C 76071,CCCCC1CNC(=O)CN1.C1(NC(=O)OC(C)(C)C)CC(F)(F)C1 76072,N1(C(C2C(NC(CCC3(C#N)CCC3)=O)CC2)=O)CC2CC1CS2=O 76073,c1(C(=O)NC(C2(O)CCN(C(C3(C)CC3C)=O)CC2)C)nn2cccnc2c1Cl 76074,C12(NC(C(CC)NC(C)=O)=O)CCC(CC1)N(C(=O)C=C1CCCCC1(C)C)C2 76075,C1(C(N2CCC(N(C)C(c3coc(C(N)=O)c3)=O)C2)=O)(OCC)CCOCC1 76076,c1(C(=O)NCC2(CNC(C(C(C)O)C)=O)CCOCC2)ccc2ccoc2c1 76077,c1(COCCNC(=O)NCC(O)C2CC2)ccco1 76078,c1(NC(C)=O)cc(C(=O)NCCNC(C2CCCOC2C)=O)ccc1F 76079,N1(c2cc(OC)nc(OC)n2)CCC2CN(C(c3cc(SC)nn3C)=O)CC2C1 76080,C1(C)(C(N2CC(OC)(CO)C2)=O)CC(O)CN1C(=O)C=C(C)C(C)C 76081,N1(C(c2c(C)nsc2)=O)CC(NC(=O)COCc2nc[nH]n2)CC1C 76082,C(C(C)C(C)N=c1nc(N2CCC(CCO)CC2)c2cc(Cl)ccc2[nH]1)OC 76083,C1(C(N2CCC(OC3CN(C(CCCOCC)=O)C3)CC2)=O)CC(C)OC(C)C1 76084,CC1CCN(C(=O)COC(=O)CO)C1CNC(=O)CCCC1CC1 76085,c1(C(CC)NC(=O)C(=O)NC(c2cccc(C)c2)C)cn2cccnc2n1 76086,C1(NC(c2c(C)cccc2F)=O)CC(C2CCN(C(=O)Cc3csc(Cl)c3)C2)C1 76087,Cc1cccc2[nH]cc(C(=O)NCCN(C(=O)C(C)n3ccnc3)CC(C)O)c12 76088,C1(OC)CC(CNC(=O)C2=CCCS2)N(C(=O)CC2(C)CCCCC2)C1 76089,C1(NC(c2cn[nH]c2)=O)CN(C(c2cncc(-n3ccnc3)n2)=O)CCC1CO 76090,N1(C(CC)=O)CCC(N=c2nc(N3CCC=CC3)c3c([nH]2)CCC(C)C3)C1 76091,N1(C(C2(C)COCCO2)=O)CC2CC(NC(c3ccn(CCF)n3)=O)C1C2 76092,c1(CCC(=O)N(CCC(C)NC(C(CC)(C)O)=O)C)nnc(O)nc1O 76093,Cc1cc(Cl)c(Br)cc1S(=O)(=O)NCCNc1ccccc1[N+](=O)[O-] 76094,c1(C(CNC(=O)CN2CCCC2=O)NC(C(C)OCC=C)=O)ccccc1F 76095,N1(C(c2nnc(C)s2)=O)CC(O)C(O)C1CNC(=O)Cc1ccc(F)cc1F 76096,n1(CC(=O)NCC2CC(C)N(C(=O)C(C3CC3)C3CC3)C2)nc(O)ccc1=O 76097,c1(C(=O)NCC2C(C)(C)CN(C(C3CC4C=CC3C4)=O)C2)nnc2ccccn12 76098,c1(CC)sccc1C(=O)NC(C1CCCN1C(c1cnco1)=O)C 76099,N1(C(C2N(C(C3CCN3CC(F)(F)F)=O)CCC2)=O)CCC(CO)C(F)C1 76100,CC1CN(C2CC2)CCN1C(=O)C(c1ccc(C2CC2)cc1)O 76101,N1(C(c2cnc(CC)nc2)=O)CCC(NC(=O)Cc2ccn(CC)n2)C12CC2 76102,c1(C(=O)NCC2CCCC2Nc2cc(C(F)(F)F)ncn2)cn2c(n1)COCC2 76103,c1(OC)ccc(C(N2CC(CO)(NC(=O)COCCSC(C)C)C2)=O)cc1Cl 76104,Cn1cc([N+](=O)[O-])c(=NCC2(F)CCN(C(c3ccc(S(C)(=O)=O)o3)=O)CC2)[nH]1 76105,c1(OC)ccc2[nH]c(=NCC(C)NC(c3cc4c(C)cc(C)nc4s3)=O)sc2n1 76106,N1(C(C2(CCOC)CC2)=O)CC2CCCC(C1)N2C(C1CCCC1S(C)(=O)=O)=O 76107,Cc1csc(=O)n1CCCC(=O)NC1CC(N(C)C(c2cc(Cl)cn2C)=O)C1 76108,N1(NCc2ncn(C)c2)CCC(NC(c2ccc3c[nH]nc3c2)=O)C(F)(F)C1 76109,C12(NC(N(CCOCC)CC)=O)CCC1CCN2 76110,c1(C(N2CC(C(C(=O)N(CCCC=C)C)OC)C2)=O)coc(N(C)C)n1 76111,c1(C(C)(C)C)ccccc1C(=O)NC12CC(CNC(C3CC3C(F)(F)F)=O)(C1)C2 76112,[N-]=[N+]=Nc1ccccc1C(=O)NC1(CF)CCN(C(=O)Cn2cccn2)C1 76113,C1(NC(C(CC)OCC)=O)CCC2CN(C(=O)C(C)Sc3ncccn3)CC2C1 76114,C1(NC(CCC(=C)C)=O)CCN(C(C2CCC(=O)C2)=O)CC(O)C1 76115,c1(CC)ccc(F)c(C(N2CCCC2(C)CNC(=O)C(C)(F)C(=O)OC)=O)c1 76116,c1(C(=O)NCC2C=CCN2C(c2sccc2C(F)F)=O)ccc(OC(F)F)nc1 76117,C#CCC(C)(C)C(=O)NCC(C1(O)CCN(C(c2ncncc2N)=O)C1)C 76118,C1(OC(c2c(C)ncnc2)=O)CCCCCCCCC1 76119,C12N(CC1(C)C)C(=O)CC1CCCC(C1)NC2=O.c1(COC)cccnn1 76120,N1(C(C2(S(N)(=O)=O)CCCC2)=O)CCC2(CC1)OCCC2NC(C1CCCC1)=O 76121,c1(C(N2C(CNC(=O)CC3CC4(CC4)C3)CCC2)=O)cc(O)ncn1 76122,C1(CCNC(c2cc(C)on2)=O)CCCCN1C(c1cc(C(N)=O)no1)=O 76123,N1(C(Cc2nc(C)[nH]n2)=O)CCCCC1CCCNC(=O)C(F)CC1CC1 76124,C(=O)(CS(=O)(=O)C(C)C)N1CC(OC)CC1(C)CNC(=O)C=Cc1ccoc1 76125,N#CC12CCCCCC1CN(c1ccn3nccc3n1)C2 76126,N1(C(c2c(CC)nnc(C)c2)=O)CC(NC(C2CN(CC)C2)=O)CC12CCOC2 76127,c1(C(=O)OCC)cnc(NC2(CNC(c3cccc(Cl)c3F)=O)CCC2)nc1C 76128,c1(-c2scc(C(=O)NC3C(CNC(C(COC)C)=O)C3)n2)ccc2c(c1)CCO2 76129,CC1(C)NC(=O)CC1C(N1CC(C(=O)NC2CCCN(O)C2=O)C(F)(F)C1)=O 76130,CC(CNC(=O)C(C)(C1CC1)N(C(=O)CC1NC(=O)NC1=O)C)C(C)(C)C 76131,Cc1cc(C(=O)NC2CN(C(=O)Cc3cscn3)CCC2F)cnc1O 76132,Cc1c(C(=O)NCC(CNC(=O)Cc2nc[nH]n2)CO)sc2nnc(S)n12 76133,C1(N(C(c2c(COC)cccc2)=O)C)CN(C(=O)CC2CC(OC)C2)CC12CC2 76134,N#CC1CCC(C(=O)NCC2CC(CNC(=O)C(c3ccccc3)O)C2)CC1 76135,C1(C(N2CCC(CC#C)CC2)=O)CN(C)CCN1C(C1C2COCC12)=O 76136,c1(CN(C(C(c2cn(C)nn2)NC(Cn2c(C)nnn2)=O)=O)C)ccccc1F 76137,C12(CC)CN(C(=O)CC(C)OC)C(CNC(=O)CC3C(=O)NN=C3C)(C1)C2 76138,N1(C(CC=CCNC(CC=C(C)C)=O)=O)CCC(COC(C)C)CC1 76139,c1(C(c2nnnn2CCSC)NCC(c2ccccc2)OCC)cscc1Br 76140,c1(CNC(c2n(C(C)C)ccn2)=O)ccc(C(=O)NCC2CSCCO2)nc1 76141,N1(C(C(C(CNC(c2ccnc(OC)n2)=O)C)F)=O)CCc2nc(O)[nH]c2C1 76142,C(N=c1cc(C(c2ccccc2)C)nc[nH]1)C1(SC)CCCCC1.C1CCCC1 76143,C1(C)(C(=O)NCC2CC(C(=O)NC(c3nc(C)on3)C)C2)CNC(=O)C1 76144,C(=O)(C(C)CS(C)(=O)=O)NCCC(C)CF 76145,CCCCCCSC1CN(C(N)=O)C1.c12nnnn1CCNC2COC(C)(C)C 76146,Cc1oc(C(C)C)nc1C(=O)NC1CCCCC1NC(=O)CNC(=O)C(C)(C)C 76147,Cc1ccnc(C(=O)N(C2CCC(NC(c3sc(Cl)cc3Cl)=O)C2)C)n1 76148,CC1C(C)N(C(c2ccc(N(C)C)cc2)=O)CCN1C(=O)CC(O)CCN(C)C 76149,Cc1cccc(NC(N2CCN(C(c3noc(C)c3C)=O)C(C)C2)=O)c1C 76150,N1(C(CN2C(=O)COCC2)=O)CCC2CCC(C1)N2C(=O)CN1CCCC1CO 76151,N1(C(C2CC(CNC(CCOCCOC)=O)OC2)=O)Cc2ncsc2C1 76152,Cc1cc2cc(C(=O)NCC3CC3CNC(C3CCC3)=O)oc2cc1C 76153,c1(C(N2C(C)CC(NC(C3CC(=C)C3)=O)C2)=O)ccc2c(c1)OCCC2 76154,c1(C(=O)NC(CC=C)CNC(C2(CSC)CCOCC2)=O)nc(OC)ccc1Cl 76155,N1(C(C)=O)CCCC1(C)C(=O)N(CCCNC(C1(CC(C)C)CC1)=O)C 76156,C12(NC(C3CCC34CCC4)=O)CCCC(CN(C(c3cnsn3)=O)C1)C2 76157,CN1C(=O)C2CN(c3cc(C#N)ncn3)CC2C1=O 76158,C1(CC=C)(C(=O)NCC(O)CNC(C2(C(N)=O)CC2)=O)CCNC1=O 76159,C1(N(CC#C)C(c2ccc(COC)o2)=O)CCN(C(=O)CCN(C)CCC)CC1 76160,CCCC(O)C(=O)N1CCC(C(=O)N(CCC)C(C)C)C1 76161,C1(CC(N2C(CNC(C3CCCC(OC)C3)=O)CC2)=O)CCn2cncc2C1 76162,N1(C(C#CC(C)C)=O)CC(NC(c2coc(Br)n2)=O)C(C2CC2)C1 76163,N1(C(c2cc3ccoc3cn2)=O)CCCC2C1CCN2c1ncc(Cl)cn1 76164,C(=O)(C1c2[nH]cnc2CCN1C(=O)C(CSC)c1ccccc1)OC 76165,C1(C(=O)NCCCCO)CN(C(=O)CC2CCOC2=O)CC12CC2 76166,C1(=CC(=O)NCCC2(NC(C(C)OCC3CC3)=O)CCCC2)CN2CCC1CC2 76167,Cc1cc(NC(=O)CC2(C)CCN2C(C2(C)CC2)=O)c([N+](=O)[O-])cc1Br 76168,CC(O)C(C(=O)N(CCCNC(=O)CCC1CCCCCC1)C)NC(=O)C1CC1 76169,C1(C(N(C(CN(C(C)=O)C)C)C)=O)CC(NC(=O)CN(C(=O)C(C)C)C)CCO1 76170,C1(NC(CC(C)N(C)C)=O)CN(C(=O)C(C)(C)n2ccc(C3CC3)n2)CCC1(C)C 76171,C1(C(N(CCCn2cc(CCCS(N)(=O)=O)nn2)C)=O)CCOC2(CCCC2)C1 76172,C1(F)(CSc2nnn(C(C)(C)C)n2)CCCOC1.C12CC1CN2 76173,N1(C(CNC(C(CC)NC(=O)OCCOC(C)(C)C)=O)=O)CCc2nc(I)[nH]c2C1 76174,C(=O)(CCN=c1nc2c(ncn2C(C)C)c(NCCCCCSC)[nH]1)NCC 76175,C=C(C)C1CCC(C)(O)C(NC(C2(c3cccc(C(F)(F)F)c3)CCC2)=O)C1 76176,c1(NC(C2(C)CCN(C(=O)Nc3ccc(C)cc3)C2)=O)csc2nccnc12 76177,C(c1cncn1C)=CC(=O)NC1CC(C(C)NC(=O)CC2CCOC2)C1 76178,C1(NC(C2CC(N(C)C)C2)=O)CCCC(NC(c2ccc(=O)oc2)=O)C1 76179,C1(C(=O)NCC(C)(C)OCC(=O)N(C2CCCC2C#N)C)CCCCCC1 76180,C(C(C)(CC(C)C)NC(c1cc(C(N)=O)on1)=O)NC(C(C)=CC1CC1)=O 76181,c1(C(N2C(CC(=O)N(C(C=C)C)C)CC2)=O)cnn2ccccc12 76182,CN=c1[nH]cc(C(N2CCC(O)(C(C)CNC(c3cn(C(C)C)nn3)=O)C2)=O)o1 76183,c1(C(=O)NCC(Cn2cc(CC(CC)(C)O)nn2)(F)F)ccc(=O)n(C(C)C)c1 76184,CC#CC1CCN(C(c2coc(CNC(=O)COCC3CCCO3)c2)=O)CC1 76185,N1(c2nccc(SC)n2)CCC(C2CN(c3cc(C)ncn3)C2)CC1 76186,N1(C(CCCCC=CC)=O)CCC(C2CCN(C(C3CC3(F)F)=O)CC2)C1 76187,N1(C(C(CC)(C)COC)=O)CCC2(C=C(C(=O)N(C3CCC3)C3CC3)C2)C1 76188,NC(=O)CCC(N)C(=O)N1C(C(=O)NC2COC(=O)C2)CC2CC12 76189,C=CCC(CC(F)F)C(=O)N1CCCOC(CCNC(=O)C(=O)C(C)(C)C)C1 76190,Cc1c(-n2nc(Cc3ccccn3)nc2CCCCS(N)(=O)=O)cccc1Cl 76191,C=C(C)CCCC(=O)N1CCCCCC1CNC(=O)CC1CCCCN1C 76192,N1(C(c2cc(C)no2)=O)CC2CC(NC(=O)C(CC(F)F)C3CCC3)C2C1 76193,c1(C(=O)Nc2ccc(C(N3C(CCC=C)CCC3)=O)nc2)cnnc(C)c1C 76194,C(=O)(C1c2c[nH]nc2CN1C(C1CCCCN1C)=O)N(CCC(=O)NC)CC 76195,C1(c2ccccc2)(NC(C2C(OC)CCC2)=O)CCN(C(c2cnsc2)=O)CC1 76196,C1(C(N2CCC(NC(=O)CC3CCCCC3)C23CC3)=O)CC2CCC(C1)C2O 76197,C1(CC=C)(C(=O)NC(C)C(N)=O)CCCN1C(c1ccc(C)cn1)=O 76198,C1(C(=O)NCC2(C)CC2)CC12CCN(Cc1cccc(Br)n1)CC2 76199,Cc1cnn(CC(=O)N(C2CCCC2)CCN(C(=O)Cc2cc(OC)no2)C)c1 76200,C1(C(=O)Nc2ccc(NC(=O)NCC)cc2)CC2CCCC2C1 76201,C1(C)(C(N(CCOC)CCn2cc(C3(CCO)CC3)nn2)=O)CC(C#N)C1 76202,c1(C(=O)NC2COCCN(C(C=CC(CC)C)=O)C2)cc2c(cn1)OCO2 76203,C#CC1(CO)COCCN1C(N1CCC(CC)(NC(=O)OC(C)(C)C)C1)=O 76204,C(=O)(CC(F)(F)C(F)(F)F)NCCC(C(C)C)NC(=O)C(=O)NCC1CC1 76205,C1(OCC(=O)NCC(=O)OC(COC)C2CCC2)CCCC1 76206,CCC(CC1CCCC1)C(=O)NC1CCCCC1NC(C1OCCCO1)=O 76207,N1(C(C)C)CCC(CC(=O)N(C)CC2CCN(C(C3C(C)C3(F)F)=O)C2)CC1 76208,C12(C(N(CC=C)CCO)=O)CCC(CC1NC(c1ncn(C)n1)=O)C2 76209,Cc1cc(C(=O)NCCN(C(=O)Cc2ccco2)C)n(C2CCC2)n1 76210,c1(C(C)C)cc(C(=O)NC2(CNC(=O)CC3CCCC34CC4)CCOC2)nn1C 76211,C(=O)(C1=C(F)CN(C(c2cscn2)=O)CC1)NC(C)CC(F)(F)F 76212,c1(NC2C(C)CN(C(=O)CCCC(=O)N(C)C)C2)ncc(Br)cc1[N+](=O)[O-] 76213,C(c1cn(C)nn1)=CC(=O)NC(C(=O)NC(CC=C)CC)CC1CC1 76214,c1(C(=O)NCC2C(CC(=O)NCc3ncsn3)C2)cc(Cl)n[nH]1 76215,N1(C(CCC2N(C)CCCC2)=O)CCCCC(CNC(c2csnn2)=O)CC1 76216,C1(C(N(CCCNC(c2ccc(C)cc2)=O)C2CC2)=O)CCC2CCC1O2 76217,N1(C(C(C)N(C)C)=O)CC2CC(NC(c3ccsn3)=O)CC1C2 76218,N1(C(C(=O)Nc2ccc(C)cc2)=O)CCCN(C(c2cc(C)c(C)cn2)=O)CC1 76219,C(=O)(CCCC(=O)N1CC(CNC(=O)CCC(=O)c2cccc(Cl)c2)C1)N(C)C 76220,Cc1cnc2cccc(C(=O)N(C(C)CNC(=O)CSCC(C)C)C)n12 76221,N1(C(c2cn(CC=C)nc2)=O)CCC2(CC2C(N2CC(C(C)OC)C2)=O)C1 76222,N1(C(C2C(=C)CC2)=O)CC(C)OC2(CCN(c3nc4cc(C)ccc4o3)CC2)C1 76223,C1(NC(Cc2n[nH]c(=NC)s2)=O)CC2CC(C1)N(C(C1(O)CCC1)=O)C2 76224,C=CCC(C)C(=O)N1CCC(C(F)F)(CNC(=O)CN(c2ccnc(Cl)n2)C)C1 76225,c1(C(N(CC(C)C)C(c2ccccc2)C)=O)cc2c3ccccc3n(C)c2s1 76226,C(CC(C)(C)C(=O)NCC(CNC(=O)C(N1CCC(O)CC1)C)OC)OC 76227,C1(C(=O)NC(c2ccccc2)C(=O)NCC(CC)C#N)CCOCC1(C)C 76228,c1(CC(=O)NCC2C(CNC(c3ncn(C)c3)=O)C2)ccc(S(N)(=O)=O)s1 76229,N1(C(C(CC)(C)O)=O)CCOCC(CNC(=O)CCc2ccn(C)n2)C1 76230,CCC(CN(C)C)CC(=O)N1CCCCC1CN(C)C(C1CCCC2(CC2)C1)=O 76231,c1(CC)cccc(C(N2CCCC(NC(C3CCC4(CCC4)C3)=O)CC2)=O)c1O 76232,CN=c1[nH]cc(-c2cnc(NCC3CCO3)c(C(=O)OC)c2)cc1C#N 76233,c1(Cn2cc(C(C=C)(C)O)nn2)ccc(CNC(c2ccc(C(F)F)o2)=O)cc1 76234,C1(N(CC(=O)NC(c2cn(C)nc2)CO)C(n2cccn2)=O)CCC(C2CC2)C1 76235,O(NC(=O)C(C)CC1CCCO1)CC(=O)Nc1cc(SC)sc1Cl 76236,C1(C(=O)NC(CC(=O)NC(C)C)C)CCCCCN1C(C1CC(=O)NC(=O)N1)=O 76237,Cc1cc(C2CC2C)nc(C(=O)NCCCOCCNC(=O)COCCOC)n1 76238,c1(C(N(C2CCN(C(C(C(C)C)OC)=O)C2)C)=O)cc([N+](=O)[O-])c(C)cc1C 76239,c1(-c2nc(-c3ccc(OC)cc3)nn2C2CC2)cnc(OC)c(Cl)c1 76240,c1(CC)ccc(C=CC(N2CC(NC(c3nc(C)no3)=O)CC2C)=O)cc1 76241,C1(CNC(C(c2ccccc2)N(C)C)=O)CC2CC2N1C(=O)C(=O)NC1CC1 76242,c1(C(=O)NC(C(C)C)C(C)NC(c2ccc(N(C)C)nc2)=O)cn(C)c(=O)n1C 76243,c1(NCC(CC(C)C)N(C)C)ncccc1S(=O)(=O)NCC12CCN(CC1)CC2 76244,C12(C(=O)NCC(C)(CNC(=O)C(C)(C)OC(C)=O)OC)CCC(F)(CC1)CC2 76245,Cc1c(C(N2CCC(N(C(=O)CSC(F)(F)F)C)C2)=O)cc(C(C)C)n1C 76246,c1(C(=O)NC(C(C)(C)C)CNC(C2C3CCCC23)=O)cnn2ccccc12 76247,c1(OC)noc(C2CC2)c1C(=O)NCCC(C)NC(=O)C(C(C)C)NS(N)(=O)=O 76248,c1(CC(=O)N(CC(=O)NCC2(C(C)(F)F)CC2)CCC)cccnc1 76249,N1(C(Cc2c(C)noc2)=O)CC(O)CCC1C(=O)NCC(C)(O)C1CCCC1 76250,CCC(C)(C(=O)OC)NC(=O)C(CNC(c1c[nH]nc1OC)=O)OC 76251,N1(C(C(C(C)C)n2cccc2)=O)CCCN(C(C2CC3(F)CC2C3)=O)CC1 76252,C1(C(=O)NC2CCC(CNC(C(C=C)(C)O)=O)C2)CCc2cncn2C1 76253,N1(C(=O)Cc2cnn(C(F)F)c2)CC2CCCC(C1)N2C(C1(O)CCC1)=O 76254,C(CNC(=O)CSCCN(C)C)(CCNC(C1CCC1(F)F)=O)OC 76255,c1(C(N(C2CN(C(c3cc(C)c(C)s3)=O)CC2O)C)=O)cc2scnc2[nH]1 76256,Cc1cn2cc(C(=O)N(C)CC3CCN(C(=O)C(C)(C)C)C3)nc2s1 76257,C1(O)(CNC(C2(C#C)CCC2)=O)CCCN(C(=O)Cc2ccccc2SC)C1 76258,c1(C(=O)NC(C(C)NC(=O)COCC2CC2)(C)C)ccc2c(c1)nc(O)n2C 76259,C(=O)(C1=CCCC1)NC1CCC(NC(c2ccc(COC)s2)=O)C1 76260,c1(C(=O)NC(CCNC(C2ON=C(C)C2)=O)C)ccc(C)c2c1CCCN2 76261,Cc1cc(N)c(Br)cc1C(=O)NCC1(C)CCCN1C(=O)C(C)CN(C)C 76262,c1(C(C)=O)ccc(C(N2CCN(C(=O)Cn3cnnn3)CC2)=O)cc1 76263,N1(C(CCC(N)=O)=O)CCN(C(C2CC2F)=O)C(c2cn[nH]c2)C1 76264,C(=O)(C(CC)C(C)C)N(CCCOC1CCN(C(C2C(CCC)C2)=O)CC1)CC 76265,c1(C(=O)NC2(C)CC(NC(=O)CC3=CCCC3)C2)cnc2ccsc2c1 76266,C(C)(CC(=O)NCC(c1cccs1)O)NC(CNC(C)=O)=O 76267,c1(C(=O)NC(C(N2CCC3(CC(F)C3)C2)=O)C2(C)CC2)ncc2ccccn12 76268,Cc1cc(=NCC(F)c2ccc(C)c(C)c2)[nH]c(NC2CCCn3ncnc32)n1 76269,C1(NC(c2ccccc2)C)CCOC1c1ccccc1 76270,C(C)(C(=O)OC(C)(C)C)(C(=O)N1CCC(N(C(=O)C(C)CSC)C)CC1)OC 76271,CCCC(C)(CCC)C(=O)NCCN1CCN(C(=O)C(C)(F)C(=O)OC)CC1 76272,C1(CC(=O)N(C2CCN(C(c3cc(C(F)(F)F)n[nH]3)=O)CC2)C)C=CS(=O)(=O)C1 76273,C1(CC(=O)N(CCCCC)C)CCCC1NC(=O)Cc1nccn1C 76274,C(=O)(CCC(C)(C)O)N1CCCC(N(C(C(CC)OCC)=O)CC)C1 76275,C1(=O)C(CC(C)C)OCNC(=O)CCN1CC=C.C1(OC)CCCCC1O 76276,Cc1c[nH]nc1C(=O)N(C(=O)CC1CSCCS1)C 76277,c1(C(N2C3C(NC(C(C)CC4CCCC4)=O)C(C3)C2)=O)c[nH]nc1S(N)(=O)=O 76278,N1(C(CCC(C)OC)=O)C2CCC1C(CNC(c1cn(C)nc1C(F)(F)F)=O)C2 76279,CC(C)C(C)C(=O)NCCCN(C(c1cccc(C2CC(F)(F)C2)c1)=O)C(C)C 76280,C1(CNC(CC(CC)(F)F)=O)Cc2ccccc2CN1C(=O)CC1CC(C)=NO1 76281,C(CS(=O)(=O)CC(=O)OCc1nnn(C)c1C(F)(F)F)OC 76282,C1(NC(=O)CCSCc2ccccn2)CCCCC1NC(C1C2CCCOC12)=O 76283,N1(C(=O)COCC2CCOCC2)CC2(CCC(CO)O2)C1.C12CC(F)(C1)NC2=O 76284,Cc1nccc(C(=O)NC(C)CC(C)NC(=O)COc2c(C)cccc2Cl)c1N 76285,c1(C(=O)OC(CCC)(C)C)ccc(C(C)C)cc1 76286,C1(NC(c2ccc(C#C)cn2)=O)(CNC(C2CCCN2C)=O)CCC(C)(C)CC1 76287,c1(C(=O)NC(c2cccnc2)C(N2C(C)(C(=O)OC)CC2)=O)n[nH]c(C)c1C 76288,c1(C(N2C(CNC(=O)CCc3ccc[nH]3)CC2)=O)cccc2[nH]ncc12 76289,N1(C(c2ccccc2)=O)C2CN(Cc3ccncc3-c3sccc3CO)CC12 76290,CCCCCCC(=O)NC1CCCC(NC(C2CCC(C3CC3)C2)=O)C1 76291,Cc1sc(Cl)nc1C(N1CCN(CCNC(C2CCC2)=O)CC1)=O 76292,N1(C(COCC(=C)C)=O)CCCC1C1CCCN1C(c1nc(=N)cc[nH]1)=O 76293,N1(C(CCCCOCC)=O)CCC2CN(C(=O)CC(O)CN(C)C)CC12 76294,N1(C(C2(C#N)CC3CC3C2)=O)C2CCC1CC(NC(=O)Cc1cc[nH]n1)C2 76295,C1(C(N(C)CC2CCCN2C(C2(CO)CCCCC2)=O)=O)CCC2(CCC2)O1 76296,C1(NC(C=CCOC)=O)CC(C(=O)NC2CCN(C)C2=O)=CC1O 76297,C1(C(N2CCC(O)C2)=O)(CC)CCCN1C(=O)C=CCOC 76298,C1(CNC(c2ccc(C)c(F)c2)=O)CCN(C(c2cnc(Cl)s2)=O)C12CCC2 76299,C1(C(c2cccs2)C)CN(C(=O)Cn2cc(-c3ccc(C)c(N)c3)nn2)CCCO1 76300,C1(C(=O)NCC(=O)NOC)(OC)CCN(C(=O)C(F)C2CCC2)C1 76301,C(=O)(C#CC1CCCO1)NC(N1CCCC(c2nccc(O)n2)C1)=O 76302,N1(C(c2cc(C)c([N+](=O)[O-])cc2)=O)CCC2CN(C(C3CC(C)OC3=O)=O)CC2CC1 76303,c1(C(C(=O)N(CCCNC(CCNC(COC)=O)=O)C(C)C)C)ccn(C)c1 76304,CCCCC(C(=O)N(C)CCOCCN(C(=O)C(n1cc(Cl)cn1)C)C)C(C)C 76305,C1(C(N2CCCC(C)(C(N)=O)C2)=O)CCC2(CN(Cc3cc(O)cc(Br)c3)C2)O1 76306,c1(C(N2CCC(NC(c3cn(CCF)nn3)=O)(CO)C2)=O)cccc2cnsc12 76307,C1(C(N2CCC(NC(C3Cc4cscc4C3)=O)C2)=O)CC2(CCC2O)C1 76308,[N-]=[N+]=NCC(F)CC(C(=O)O)NC(=O)C=Cc1cn[nH]c1 76309,C=CC1CN(C(=O)CNC(=O)C2CC2)CC1NC(=O)Cn1cc(CC)cn1 76310,C1(C(=O)Nc2c(CC)cccc2)CC12CCN(S(=O)(=O)Cc1ccc(Cl)cc1)C2 76311,c1(C(=O)NC(CC(C)NC(Cc2nnc(C)o2)=O)C)ccc2nc[nH]c2c1 76312,C1(CNC(c2cn(CCO)nn2)=O)CC2CC1CN2C(c1cc(Br)c[nH]1)=O 76313,c1(C(N2CCC(NC(C(C3CC3)SC)=O)CC2C)=O)cc(S(N)(=O)=O)oc1C 76314,C(CC(C)(C)C(=O)N1CCC(O)(CCNC(=O)C(F)C2CCOC2)CC1)OC 76315,C(=O)(CC1CCc2ccccc21)N1CC2C(NC(CSc3cn(C)nc3)=O)(C2)C1 76316,C(=O)(CC1COc2cc(O)ccc21)NC1CC(CNC(C2CN(C(N)=O)C2)=O)C1 76317,n1(C(C=C)C)nc(CCOC2CCCCC2)nc1-c1cc(C(C)C)on1 76318,c1(C(=O)NCC(CC)NC(c2nc(Cl)oc2C)=O)cc(C)n(C(C)CC)n1 76319,C(=O)(C(C)(C)CC(C)C)NCCN(C(=O)CCCSc1ccc(Cl)cc1)CCC 76320,C=CCC(F)(F)C(=O)NC(CNC(c1ncc(F)cc1F)=O)C(C)C 76321,c1(C(=O)NCC(C)CNC(c2c[nH]nc2C2CCCO2)=O)cnn(C)c1C(C)C 76322,N1(C(C(C2CC2)OC)=O)CCC(C)N(C(c2cc3ccsc3s2)=O)CC1 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76515,c1(C(=O)NCC(n2cc(COCC(=O)N(C)C)nn2)C)cc(Cl)cc(Cl)c1F 76516,C1(C)(COC)CCN(C(N2CCN(C(C#N)C(C)C)CC2)=O)C1 76517,N#Cc1c(CCCNC(C2CCC3CC3CC2)=O)[nH][nH]c1=N 76518,CC1(CNC(c2cn(C(F)F)nc2C)=O)CCCN(C(C2CC23CCOC3)=O)C1 76519,C1(C(=O)NCCN(C(C2CC2(c2ccccc2)F)=O)CC)CC(S(C)(=O)=O)C1 76520,c1(CN2CC(C(=O)NCCCOC=C)SCC2)c(F)cc(O)cc1F 76521,c1(C(=O)NC2CCN(C(C=Cc3ccc(C)o3)=O)C23CC3)ccn2ncccc12 76522,C(c1cccc(C)c1)=CC(=O)NC(CCOCC)C(=O)NCCC1CC=CC1 76523,C1(CNC(c2c(SC)ccs2)=O)CCN(c2ncc(Cl)c(C(C)=O)n2)CC1C 76524,C1(C(N2CCC(C(CC)CC)C2)=O)C=CCN(C(=O)CN(C)CC)C1 76525,c1(CC)onc(-c2ccccc2)c1C(=O)NC1CCCC1NC(=O)C=CBr 76526,C1(CNC(C2(C)CC2Br)=O)CCC2(CCN(C(=O)CN=S(C)(C)=O)CC2)CO1 76527,C1(CNC(C2N(CC)CC2)=O)CN(C(C2OCCO2)=O)CC1C(F)(F)F 76528,N1(C(c2sc(C(=O)OC)c(N)c2)=O)CCN(C(c2cc(OC)ncn2)=O)C(C)C1 76529,C1(C(N2CC(C)(NC(C3N(CC)C(=O)CC3)=O)C2)=O)OCCOC1(C)C 76530,CCC(C)(COC(C)=O)CNC(=O)NCCOC(F)F 76531,N1(C(C2(O)C(C)(C)OCC2)=O)CCC(C(=O)N2CCCC(C(N)=O)C2)=C(F)C1 76532,C1(NC(C#C)=O)CCC2(C1)CN(C(C1(C#N)CCC1)=O)C2 76533,N1(C(C)C)CCOC(C(=O)NC23CC(CNC(=O)CC4CCCOCC4)(C2)C3)C1 76534,N1(C(c2cc(OC)nn2C)=O)CCN(C(c2cccc(OC(F)F)c2)=O)C2CC12 76535,c1(C(=O)NC2(CCNC(=O)C(O)C(F)F)CC2)nccn2ccnc12 76536,C(N=c1[nH]c(N2CCOC(C)(C(F)(F)F)C2)nc2cc[nH]c12)c1c(C)nccc1 76537,CP(C)(=O)CC(=O)NC1CC(CC(=O)NCc2cc(C(N)=O)co2)C1 76538,CC(=O)C1=C(c2ccc(F)cc2)N(C2CC2)C(=O)NC1c1cnc(Cl)c(F)c1 76539,C1(C(=O)NCC(=C)F)CCN(C(=O)C2=NNC(=O)C2)C(CC)C1 76540,Cc1ccccc1CC(CNC(=O)C(F)(F)C1(O)CCC1)CO 76541,c1(C(=O)NC(C(C(C)C)NC(c2cc(O)cs2)=O)C)ccc2ccn(C)c2c1 76542,C1(NC(C2CCCCC2)=O)CCN(C(C23CCCC2C3)=O)CC1O 76543,C1(CC)CN(C(c2csc(O)n2)=O)CCN1C(c1cn(C2CCCC2O)nn1)=O 76544,Cc1cc(C(=O)NC2(CCNC(=O)C=Cc3cn(C)cn3)CC2)cc(=O)n1C 76545,Cc1noc2nc(C(=O)N(C3CCN(C(=O)C(F)=C4CCC4)C3)CCO)ccc12 76546,C(C(CC(=O)N1CC(C)(C)CC1CNC(c1ncccc1O)=O)C(F)F)N(C)C 76547,C#CCC(O)C(=O)N1CC(F)(CNC(c2ccc(-c3ccccn3)s2)=O)C1 76548,CC1(NS(=O)(=O)CCCn2cnnn2)CCCNC1 76549,CN1CCCC(C)(C(=O)NC2COCCC2NC(=O)COc2ccccc2)C1 76550,N1(C(C(c2ccccc2)NC(C2=C(C)CC2)=O)=O)CC2CCC2(C)C1 76551,C1(NC(C(Cc2cn[nH]c2)NC(c2n[nH]cc2Cl)=O)=O)C=CCCCC1 76552,c1(OC)ccc2cc(C(=O)NC3CCN(C(c4cnc[nH]4)=O)C3(C)C)sc2c1 76553,N1(CC)C(=O)COC(CNC(C)C(=O)Nc2ccc(Br)cc2)C1c1nccn1C 76554,N1(C(CN(CCOC)C)=O)CC2(CC(NC(=O)CCSC)c3nccn32)C1 76555,C1(O)(C(=O)NCC2CN(C(c3scc(C)c3Br)=O)C2)CCCCCC1 76556,c1(CNC(=O)CC2OCCCO2)cc(C2CCCC2)ccn1 76557,CCC(C(=O)NC1CC(F)CN(C(c2cc(C(F)F)cs2)=O)C1)C(C)C 76558,S(=O)(=O)(c1cc(Br)c(Br)s1)Nc1nc(C(=O)NC(c2ccno2)C)n(C)c1 76559,N1(C(C(CC)(O)c2ccccc2)=O)CCC(NC(=O)CC(=O)NC2CC2)C(F)C1 76560,n1(CC(C(=O)NC(CNC(c2scc(NC)n2)=O)CO)C)nnc2ccccc12 76561,CN1CC(NC(C2CCCC(NC(c3ccc(C#N)o3)=O)CC2)=O)C(F)(F)C1 76562,Cc1ccc(C(C)C(=O)N(CC(O)CNC(c2csc(Br)n2)=O)C)s1 76563,C(=O)(CC(C(F)(F)F)n1ccnc1)NCC(=O)NCCCC(N)=O 76564,C1(C(N(CCCN(C(=O)CC2C=CCCC2)C)C)=O)C2CCC1(c1ccco1)C2 76565,c1(C(=O)NCC2CN(S(=O)(=O)CCCCl)CCO2)ccc2c(c1)CCO2 76566,C(=O)(CC(=O)N1CCC1CNC(C1CCCCO1)=O)NCC#C 76567,c1(-n2c(C(C3CCC3)O)nc(CCCC)n2)ccc(Br)cc1OC 76568,N1(C(c2coc(Cl)n2)=O)CC2(CCCN2C(c2ccc(CO)cc2)=O)C1 76569,CC(C)CC(CC(C)C)C(=O)NCCN(C1CCCCC1)C(C1CCC(O)C1)=O 76570,N1(CC(=O)NCC(C)N(C)C(C2(SC3CCCCO3)CC2)=O)CCN(C)CC1 76571,c1(C(C)NC(C2C(CNC(C3(SC)CC(=O)C3)=O)CCC2)=O)ccc(C)nc1 76572,N1(C(=O)Cn2cncn2)CCC2(CC1)CC2NC(C1(C2OCCO2)CC1)=O 76573,C12(COC)CC(NC(=O)CNC=O)(CN1C(=O)CCc1ccccc1OC)C2 76574,C1(NC(C2N(CC)CC2)=O)CCCN(c2nccc(-c3ccc(F)cc3)n2)C1C 76575,C12(NC(CCc3c(C)noc3Cl)=O)CCC(CN(C(=O)C(C)C(C)(C)C)C1)C2 76576,c1(C(=O)NCC(CC)(CC)NC(c2ccnc(C)n2)=O)ccc2nc(S)[nH]c2c1 76577,N1(C(C2(NC(CCC(=O)NC)=O)CC2C)=O)CCCC(C)(N(C)C)C1 76578,c1(C(C)C)nocc1C(=O)N(C(C)CNCc1ccnn1C)C 76579,c1(OC)ccc(Br)c(C)c1C(N1CC(C)(CNC(c2oncc2C)=O)C1)=O 76580,C(c1cc(OC(C)C#N)cc(OC)c1)=CC(N1CC(CC(=O)OCC)C(O)C1)=O 76581,CC(C)C(O)C(C)C(=O)NCCC(C)(C)NC(c1ccncc1Br)=O 76582,C(=O)(CCC(=O)NCCC1CCCN1C(C1CCCSC1C)=O)NC 76583,C(=O)(C1=C(Cl)CCCC1)NCC1C(NC(COCc2n(C)ccn2)=O)CC1 76584,Cc1ncc(CC(=O)NC2(CNC(c3ccccc3C)=O)CC2)c(O)n1 76585,Cc1cc(CC(=O)NCC(C)(C)CN(C(=O)CCC2CCC(C)O2)C)ccc1Cl 76586,c1(C(C)(C)C(=O)NCC2C3CN(C(C4CC4CF)=O)CC23)nccn2cnnc12 76587,c1(C(=O)NC(CC)CNC(=O)CC2(C)CC2(Cl)Cl)cnn2c(=N)[nH]cnc12 76588,C1(CN(C2CCN(Cc3ccccc3)C2)C)CCCCN1C(=O)CCCC1CC1 76589,C1(O)(CNC(C2CCC2)=O)CCN(C(c2ccc(-c3ncc[nH]3)cc2)=O)C1 76590,N1(C(C2(COC)CC2)=O)CCN(C(=O)CN(C)C(c2[nH]cnc2C)=O)CC1 76591,N1(C(c2nccc(C)c2O)=O)CCN(C(c2ccc(Cl)o2)=O)C(C)C1C 76592,c1(CC(=O)OC)cscc1C(=O)NC(C)C(C)NC(c1ccsc1)=O 76593,c1(-c2n(C)ncc2)cccc(NC(=O)CN2CCC(N3CCNC(=O)C3)CC2)c1 76594,c1(C(=O)OC)cc2cc(C(N3CCN(C(=O)C(C(C)C)N(C)C)CC3)=O)sc2[nH]1 76595,N1(C(C=Cc2c(C)noc2C)=O)CC2CCC1CN2C(=O)Cc1sccc1Cl 76596,C(=O)(CCC(CF)CF)NC1CC2CC(NC(=O)C=CCF)C2C1 76597,c1(C(N2CCN(C(c3ccc(CC(F)F)cc3)=O)CC2)=O)c[nH]c2ccccc12 76598,c1(C(C(=O)NCC2(O)CN(C(C(CC)N(C)C)=O)C2)CC)ccc(F)cc1 76599,c1(C2CCN(CC(=O)NC)CC2)ccc(C(=O)OC)cc1OC.C1(=O)C=CO1 76600,C(=O)(CCC(N)=O)N1C(C(C)NC(c2cnoc2C2CC2)=O)CCC1 76601,c1(C(=O)NC2(CO)CCCN(C(CN(CCOC)C)=O)C2)ccn2cccc2c1 76602,N1(C(c2cc(OC)c(F)cc2)=O)CCc2sc(-c3ccc(C(C)N)cc3)nc2C1 76603,C1(NC(CN(C(C(C)C)=O)C)=O)C(C)CN(C(=O)CCCn2cncn2)CC1C 76604,N1(C(c2nc(C(=O)OC)oc2)=O)CCCCC(NC(=O)Cc2nocc2C)C1 76605,c1(C(N2CCC(O)(CCNC(c3ccc(Cl)s3)=O)C2)=O)cnc(C2CC2)nc1O 76606,CC1CCC(NC(=O)CC2CS(=O)(=O)C2)CN1C(=O)CNC(N1CCCC1)=O 76607,N1(C(CCSCC)=O)CCC(C(=O)NCC2CC(O)C23CCC3)CC1CC 76608,C#CCCCCCC(=O)NCc1nc(C(N2CCOC(CC)C2)=O)c(C)o1 76609,C1(NC(C2(CC)CCCN2C(=O)CC(C)COC)=O)CC2(CCOC2)C1 76610,N1(C(C2(C(F)(F)F)CCN(C)C2)=O)CCC(NC(c2cccnc2)=O)C(C)(C)C1 76611,c1(NC(CNC(c2nn(CC)c(C)c2)=O)(C)Cn2cccn2)snc(C)c1C#N 76612,c1(C(N2CCN(CC(=O)NCC3(C)CCCC3O)CC2)=O)ncn2c1CCC2 76613,C(=O)(C(CN=[N+]=[N-])NC(=O)C(C)NC=O)NC1(c2nc(C)[nH]n2)CC1 76614,C=CCCC(C(=O)NC1CN(C)CC1(C)C)NC(=O)C(n1ccc(C)n1)C 76615,c1(C(N2C(CCNC(Cc3c(C)nsc3)=O)CCC2)=O)cnc2c(c1)OCCN2 76616,CCC(O)(CNC(=O)Nc1ccc(F)nc1)CCC(F)(F)F 76617,CC(CN=c1[nH]c(=NC2COC(C3CC3)C2)[nH]c2ccsc12)c1cccs1 76618,N1(C(C(C)(C)SC)=O)CCC(NC(C2(C)CC2(F)F)=O)C(CO)CC1 76619,C(=O)(C(C)C(O)C(C)C)NC12CC(NC(c3cc(C(C)C)on3)=O)C(OC1)C2 76620,C(=O)(C(C)C(O)C(C)C)N(CCC(=O)NCCOCC)CC 76621,C(C)(CCCC(=O)NCCCc1nccs1)NC(C(C)NC(CC)(C)C)=O 76622,C1(C(N(CC(C)NC(CCOC)=O)C)=O)CC(Br)(Br)C1 76623,CCC(C)C(O)C(=O)NC1CCC(CNC(c2cccnc2N2CCCC2)=O)C1 76624,C1(OC)CN(C(C2C(C)(C)C2(F)F)=O)CC1NC(c1cc(C)c(C)s1)=O 76625,c1(CCC(=O)NCCN2CCC(NC(C3CC4CCC34)=O)CC2)ccccc1O 76626,c1(C(=O)NC2CCC(C)N(C(C3CSCCS3)=O)C2)cnc2c(c1)C(=O)CCC2 76627,C=C1CCCN(C(C2CC2C(C)NC(c2coc(CCC)n2)=O)=O)C1 76628,C12(C(=O)NCc3ccc(CNC(C(C)C)=O)cc3F)CCOC1CCOC2 76629,C(CCN(C)C(c1cccc(N(C)C)c1)=O)(C(C)C)NC(C(COC)N(C)C)=O 76630,c1(NC(N(C(C)C(=O)N(C2CCOC2)C)C)=O)nnn(C)n1 76631,C(CCSC)(CN=c1[nH]c(C)cc(=NCCNC(c2cccnc2)=O)[nH]1)OC 76632,NC(=O)CC(O)C(=O)N1CCCC(CCNC(c2c[nH]nc2C2CC2)=O)CC1 76633,C1(OCCNCCCC=C)CCC(CCC)CC1 76634,CC(C)CC(CN=c1[nH]c(C2CC2)nc2c1CCC2)NC(c1cnc(Cl)s1)=O 76635,N#Cc1cc(S(=O)(=O)N2CC3CCN(Cc4cc(Br)cs4)CC3C2)ccc1Br 76636,C1(O)(CNC(c2c(SC)cccn2)=O)CCCN(C(C2(O)CCCCCC2)=O)C1 76637,CC1CCC(C(N2CCC(C(C)NC(C3CC4CCC(C3)C4)=O)CC2)=O)CC1C 76638,C12(NC(Cc3cn(C)nc3)=O)CCCC1N(C(c1coc3c1COC3)=O)CCC2 76639,C(=O)(C(C)(C)CCCOC)N(CCNC(c1nn(CC)nc1C)=O)C1CC1 76640,C1(CC(=O)N(CCCC(C)C)C)CC2(C1)CN(C(=O)C(O)C1CCC1)C2 76641,Cc1noc(C)c1S(=O)(=O)NCCCNC(c1c(N)ccc(F)c1F)=O 76642,c1(C(=O)NCCNC(=O)CNC(=O)NC2CC2F)ccccc1F 76643,c1(CCC(=O)NCC(n2cc(CCN(C)CC)nn2)C)nnc(C)n1C 76644,c1(C(=O)NC2CN(C(c3scc(C)c3)=O)C3C2C3)c(F)ccc2n[nH]cc12 76645,C#CCC(C)(CC)C(=O)NCCC1CN(C(=O)C=Cc2c(C)coc2C)CCO1 76646,C(=O)(C1=CNS(=O)(=O)N=C1C)NC1C(CNC(C2(COC)CCCCO2)=O)CC1 76647,N1(C(C(C)CO)=O)CCCC(C)(C)C1C(=O)NCC(C)(C)N(C)C1CC1 76648,N#Cc1cccc(F)c1CC(N1CC2CC(NC(C3CC34CCCC4)=O)C1C2)=O 76649,c1(C(=O)NC2CN(C(C)=O)CC2c2cnn(C)c2)cc(N=S(C)(C)=O)ccn1 76650,Cc1ccc(C(=O)NCC2CC(NC(=O)C(C)Cn3ccnc3)C2)cc1Br 76651,C1(CNC(CC2C(C)CCC2)=O)CC2(CC2)CN1C(=O)Cn1ncc(O)nc1=O 76652,c1(CN(C(C#CCNC(C2C(=C)C2C(=O)OC)=O)=O)C)ccncc1C 76653,C1(CNC(c2[nH]c(=N)sc2)c2nnnn2CC2CCCO2)CCCC2(CCC2)O1 76654,N1(C(c2ccc(CC)s2)=O)CCC(N(C)C(c2ccnc(C)n2)=O)CC1 76655,c1(C(=O)NCC(C)CN(C)C(c2nccn2C)=O)ccc(F)c2c1CCC2 76656,c1(C(c2nnnn2CC2CC2)NCC=CCOC)ccc(C(F)(F)F)s1 76657,Cc1n[nH]c(C)c1CCNC(=O)C(C)N(C(C1CCN(C(N)=O)C1)=O)C1CC1 76658,N1(C(C(CC)O)=O)CCC2(C=C(C(=O)N3CC(N4CCC4)C3)C2)C1 76659,c1(C(N2CCC3(CC3C(N3CC(O)(CO)C3)=O)C2)=O)cccc2c1CCC2 76660,C#CCC(C(=O)OC)NC(=O)CCC1CCCN1C(c1cnn(CC2CC2)c1)=O 76661,C1(CNC(C2(C)CCCC2O)=O)CC2CCC1N2C(=O)Cn1cncn1 76662,C(=O)(C(CNC(=O)C(C)CCOC)C(C)(C)C)NC(c1nn[nH]n1)CC 76663,C1(C(N2CC=CC(NC(CCc3cn(C)nc3)=O)C2)=O)CSC2(C)CCC(=O)N12 76664,c1(C(=O)NCC(CNC(CC(C)C2CC2)=O)F)ccncc1Cl 76665,Cc1cc(CCC(=O)NCCCCNC(=O)C(C)c2ccsc2)ccc1Cl 76666,O=S(=O)(c1ccc(Br)cc1N1CCC2(CCSC2)C1)NCCCc1ccccn1 76667,c1(C(N2CC3=C(CN(C(C=CC(=O)O)=O)C3)C2)=O)csc2c(Cl)cccc12 76668,CCCCC(CCCC)C(=O)N1CCC(CF)(NC(=O)C=C(Cl)Cl)C1 76669,Cc1ccc(COCCC(=O)NCC2CN(C(=O)CCSC(=N)N)CCO2)cc1 76670,C1(C)(C(=O)NC(C)(C)CF)C=CCN1C(=O)CC1OCCO1 76671,S(=O)(=O)(CC(=O)N1CCCC1CCCNC(C1CC2(CSC2)C1)=O)N(CC)CC 76672,O=C(N=c1[nH]nc2cccc(Cl)n12)N1CCc2cc([N+](=O)[O-])ccc21 76673,C1(CNC(CCc2onc(C(C)C)n2)=O)CCCCN(C(c2coc(Br)c2)=O)C1 76674,C1(CCNC(C2(C#C)CC2)=O)C(C)CCCN1C(c1cccc(NC(C)C)c1)=O 76675,C1(NC(C(CC)N(CC)CC)=O)CN(C(=O)CC2COCCOC2)CCC1F 76676,C1(C(N(C2CCCN(C(=O)CCc3cnn[nH]3)C2)CC)=O)CCNC(=O)C1 76677,c1(OC)ccc(C=CC(=O)NCC(Cn2cc(C3CC3)nn2)OC)cc1Cl.CCO 76678,c1(C(=O)NCC(CC)(C)NC(c2cc3ncccc3s2)=O)cncc([N+](=O)[O-])c1 76679,c1(NC(=O)C(=O)NC2CCCCC2F)c[nH]cc(Br)c1=O 76680,N#Cc1ccc(F)c(CN2CCC(NC(c3cnn4cccc4c3)=O)CC2)c1 76681,C=CCC(CC(=O)N(C1CC2CC2C1)C)NC(=O)C(O)c1ccco1 76682,C1(NC(C(C)C2CCCO2)=O)C2CC(NC(=O)CP(C)(C)=O)CC12 76683,N1(C(C2CC(C#N)(O)C2)=O)CC2CC(NC(=O)C(c3ccc(F)cc3)F)CC2C1 76684,C1(NC(C(CC)CN(C)C)=O)COCCN(C(C2CN(C)CCN2C)=O)C1 76685,c1(C(C(=O)NCC(C)(C(C)C)NC(c2c(C)csc2)=O)C)c(C)nn(C)c1C 76686,c1(C(=O)NCCCN(C(C2CCC(C)S2)=O)CC)ccc2c(c1)NC(=O)CCC2 76687,N1(Cc2ccc(C)nc2)CCC(O)C(C(N2CC3C(C(=O)O)C3C2)=O)C1 76688,C=CC(C)(CCOC)C(=O)N1CCOC(CN(C)C(C2CC(O)(C#N)C2)=O)C1 76689,C1(CNC(C(c2ccn(C)n2)C)=O)CC(C)N(C(=O)CC2CC3(CCC3)C2)C1 76690,c1(C(N2CC(NC(C(C3CCCOC3)OC)=O)(CO)C2)=O)ccc(N(C)C)cn1 76691,C12(NC(c3ccc(O)nn3)=O)CC(C1)N(C(c1cncc(F)c1)=O)C2 76692,C(CC(C(C)(C)C)NC(c1nsnc1O)=O)N(C(Cc1ncc(C)s1)=O)C 76693,N1(C(c2occ(C)c2C)=O)CC2CCOC2(CNC(c2c(C)ncnc2O)=O)C1 76694,C1(C(=O)NC(CC)C(C)C)C=CCN(C(c2ccn(CC)c2C)=O)C1 76695,C1(O)(C(=O)NCc2c(C(=O)NCc3c(C)noc3)n(C)nn2)CCC(C)CC1 76696,N1(C(c2cccc(C)n2)=O)CCCC12CCN(C(C1CCCSC1)=O)C2 76697,C1(NC(CC(C)(C)F)=O)CC2CCC(C1)N2C(c1ccc(Cl)c(N)c1)=O 76698,C(CCCCCNC(=O)C(C)(C)CNC(C1C=CCC1)=O)OC 76699,Cn1c(C(N2CC3CC(NC(C4(C(C)(C)O)CC4)=O)CC2C3)=O)cnc1[N+](=O)[O-] 76700,O=C(C#CC1CCOC1)NCC(c1ccccc1Br)NC(CC(O)CO)=O 76701,c1(NC(C2(F)CN(Cc3cc(F)ccc3I)C2)=O)cc(Cl)nc(Cl)c1 76702,c1(OC)cccc(F)c1C(=O)NCC1CCC(NC(c2cnoc2C)=O)CC1 76703,c1(C(N2CCCC(C)(NC(C3C(OC)CCC3)=O)C2)=O)cc(O)cc(F)c1F 76704,CC1CC(NC(C2CC3CC(=O)C2O3)=O)CCN1C(=O)COCCN(C)C 76705,C1(N(C(=O)Cc2cnccn2)C)CC2CCC(C1)N2C(=O)Cc1nn(C)cc1Cl 76706,N1(C(Cc2scc(C)c2)=O)CCCC(C2CCN(c3cncc(Cl)n3)CC2)C1 76707,C1(C(N(C2CN(C(C3CC(=O)OC3(C)C)=O)C2)C)=O)CCCCC12OCCO2 76708,C1(C(=O)NC2CCC(CC)CC2)CCC2(CN(Cc3cnc(Cl)s3)C2)O1 76709,N1(C(c2c(C)nsc2C)=O)CC2(CCNC(C3(F)CCCOC3)=O)CCC1CC2 76710,c1(CC(N2CC=CC(NC(c3ccn(C(CC)CC)n3)=O)C2)=O)c(C)cccc1C 76711,Cc1nn(C)cc1CCC(N1CC2C(NC(C3(C)CC3(Cl)Cl)=O)C2C1)=O 76712,C1(CC(=O)NC(C)CN2CCCC2)CCN(C(=O)C(C)OC(C)(C)C)C12CCC2 76713,c1(C(=O)Nc2nc(C)sc2)ccc(-c2ccc(C(F)F)nc2)c2cc[nH]c12 76714,c1(C(=O)NC(C(C)C)CCN(C(=O)CC(C)(C)F)C)cccc2nc(O)n(C)c12 76715,n1(CC)cc(C(=O)NCC(O)CCNC(c2cnc(C(C)(C)C)[nH]2)=O)c(C)n1 76716,CCCC(CC)C(=O)N1CC=CC1(C)C(=O)NC1(CCC)CCC1 76717,c1(C(N2CC(CNc3cnc(-c4cccs4)s3)C2)=O)ccc(OC(F)F)c(F)c1 76718,C#Cc1ccc(C(=O)NC2CC(CO)N(C(c3ccnnc3C)=O)C2)c(F)c1Cl 76719,C1(NC(C=C(CC)CC)=O)CC2CCC1N2C(c1nn[nH]c1C(F)(F)F)=O 76720,CC(CNC(=O)CC1(NC(C2CCS(=O)(=O)N2)=O)CCCCC1)CCCO 76721,c1(C(N(CCCN(C(=O)CCC(F)F)C)C)=O)cnc2ccoc2c1 76722,C1(CNC(C(C)SC(F)(F)F)=O)CC2CN(C(=O)C=Cc3ccc(Cl)s3)CC12 76723,c1(C(=O)OC)cc(C)c(C(N2CCCCC2C2CCCN(C(=O)C(C)C)C2)=O)o1 76724,c1(NC(C(CC2CCCC2)NC(CC(C)(C)O)=O)=O)ccc(O)c(CO)c1 76725,C1(N(C(=O)C2CC2)CC)CCN(C(=O)CCCNC(c2ocnc2C)=O)CC1 76726,c1(NC(C2C(C(=O)Nc3cc(F)c(OC)c(F)c3)C2)=O)nc2cc(Br)cnc2[nH]1 76727,C1(C(=O)NCCN(C(C(C=C)O)=O)CCOCCO)CC2(CCOCC2)CO1 76728,ClCCCN=C(NCC1CCCN1c1ccccc1)NC1CCCCC12CCC2 76729,C(CC(CO)NC(=O)CC1CC(NC(C2CC2c2cccs2)=O)C1)SC 76730,N1(C(=O)COC2CCOC2)CC(C2CC2C(=O)N(CC2CC2)CC2CC2)C1 76731,Cc1cc2c(=O)n(Cc3ccc(OCC(F)(F)F)nn3)cnc2s1 76732,C1(N(C(C(C)N(CC(=O)NCC2CC2)CCC)=O)CC2CC2)COCC1(C)C 76733,Cc1cn2c(C(N3CC4(C3)CN(C(C3(C)CS(=O)(=O)C3)=O)C4)=O)c(C)nc2s1 76734,CCCC(C(=O)NC(C)CC(=O)NCC1(Cl)CC1(F)F)NC(N)=O 76735,N1(C(C2C=CC(NC(C(C)c3ccccc3)=O)C2)=O)CCCC12CCNC2=O 76736,C#CCC(O)C(=O)NCC1(CN(C)C(c2cscc2Cl)=O)CC1 76737,c1(C(=O)NC(c2ccccc2)CCC)sc(NC(c2occc2Br)=O)nc1C 76738,N1(C(C(=O)NC2C(N3CCC(C)(C)CC3)CCC2)=O)CCCC(O)(C(F)F)CC1 76739,Cc1cc(CCC(=O)NCC2CC(NC(=O)C(F)C(F)(F)F)C2)ccc1Cl 76740,c1(OC)cnc(C(=O)NCCNC(C2CC(=O)CCO2)=O)cn1 76741,CC1CN(C(=O)OC(C)(C)C)CC(NC(=O)C(CO)Oc2cn(C)cn2)O1 76742,N1(C(C(F)=CC)=O)CCCC(O)(CN(C(=O)C(C)(C)CC)C)C1 76743,C(=O)(C(C(C)C)OC)NCCOCCC(=O)N(CCCCC=C)C 76744,c1(C(N2C(C(N(C(C(=O)OC)C)C)=O)CC2C)=O)cc(C)ncn1 76745,C1(NC(c2cc(C)nc(C)n2)=O)CCC12CCCN(C(=O)C=CC1CCCC1)C2 76746,c1(C(=O)NC2CN(C(C3(CCC=C)CC3)=O)CC2F)cccc2c1C(F)(F)CC2 76747,C(Cc1cccs1)(C(=O)N=S(C)(=O)CCN)NCc1c(OC)cccc1 76748,C(=O)(CCCN(C)N=O)N1CC(COC)(CNC(=O)C(C)C(C)C)C1 76749,N1(C(COCCOCC)=O)CCCC(O)(CCNC(c2c[nH]c(=N)cc2C)=O)C1 76750,C1(NC(C(CCCOC)C)=O)CC2CCC(C1)N2C(c1cc2occc2s1)=O 76751,C1(C(=O)NCCN(c2cnc(C#N)cn2)CC)CS(=O)(=O)CC(=O)N1 76752,Cc1ccnn1CC(N1CCC(C2CCCN2C(c2ccc(Br)o2)=O)C1)=O 76753,N1(C(CC2N(C)CCC2)=O)CC2(CCCC2NC(c2cn3ncccc3n2)=O)C1 76754,c12cc(ccc1F)C(=O)NC2.C(C)(C(C)(C)SC)NC(=O)CSC(C)(C)C 76755,C(=O)(CS(=O)(=O)C(C)C)NC(C(C)NC(c1n(OC)cnc1C)=O)CO 76756,CCCCCCC(=O)N(C1CCCN(C(c2c(CC)cnn2CCO)=O)CC1)C 76757,N1(C(C(C2CCC2)OCC)=O)CCN(C(c2n[nH]c(C)c2C)=O)CC1 76758,Cc1cc(NCC2CCC2(F)F)ncc1S(=O)(=O)NC(CO)C1CC1 76759,c1(CC)cc(CN2CCN(C(=O)Nc3cccc(C)c3F)C(CC)C2)ccc1F 76760,C1(NCc2c3nc(C)oc3ccc2)CC2CC3(CC2C1)OCCO3 76761,C1(=CCNC(C(C2CCC(=O)N2)C)=O)CCN(C(=O)CCF)CC1 76762,C12(C(=O)Nc3cncc(C#C)c3)CCCC1N(C(=O)CN1CCNC1=O)CC2 76763,n1(CC(=O)NCCNC(c2cnccn2)=O)ncc2cc(Br)cnc2c1=O 76764,C(=O)(CC(C(F)F)NC(=O)CC1(NC(C)=O)CC1)NCC(=C)C(F)(F)F 76765,Cc1c(C(=O)NC(C)(C)CCNC(C2(C)CCCC2O)=O)cnn1CCC#N 76766,C1(NC(=O)CCN2CCCC2)CC2C1CCN2C(C1CCOC(=O)CC1)=O 76767,c1(C(N2C(C(=O)NCCC3CC(C)C3)CCC2C2CC2)=O)cccc2c1CCC2 76768,C1(C(C)C)(CO)CCN(C(C2CC(C)N(C(=O)CSCCC#N)C2)=O)C1 76769,C1(CNC(CC=C)=O)CCC(NC(C2(CO)CC(F)C2)=O)CC1 76770,C(=O)(C1c2ccccc2C2CC1C2)NCC1CC(NC(C=C(C)Cl)=O)C1 76771,Cc1ccc(-c2csc(C(=O)Nc3ccnc(OC(F)F)c3)c2)c(F)c1 76772,c1(NCCN(C(=O)OC)C)nc(NC(C2CCCCC2)CO)c2c(ncn2C)c1 76773,CC(O)C(C)(C)C(=O)N1CCN(C(=O)CC(O)Cc2ccccc2)CC1 76774,CC1(CNC(c2cc3occc3s2)=O)CCCN(C(C2C(F)(F)C23CC3)=O)C1 76775,c1(C(=O)OC)cc(Cl)cnc1N1CCC(C2NC(=O)NC2=O)C1 76776,c1(OC)cc(N(C)C)ccc1C(=O)NCC(C)(C(C)C)NC(=O)CC1CCOC1 76777,c1(CC(=O)NCC#CCNC(C2CCC(C)C2)=O)cc(Cl)ccc1[N+](=O)[O-] 76778,N1(C(c2c(C)nc(O)nc2C)=O)CCC2(CCOC2)C(CNC(=O)CNC=O)C1 76779,C1(C(N2CC(NC(C)=O)C2)=O)CC12CCN(C(=O)CCc1ccccc1)C2 76780,CC1(C)OC(=O)NC1C(=O)NCC1CC(NC(=O)COc2ccc(C#N)cc2)C1 76781,C1(C2CC2)(CNC(CC2C(C)(C)CCCC2)=O)CCN(C(C2SCCCS2)=O)C1 76782,c1(OC)ccc(C(=O)NC2CN(C(=O)CCCCN(C)C)CC2C)c2[nH]ncc12 76783,c1(CC(=O)NCC(CNC(=O)CC2CCOC2)OC)ccc(C)c(Cl)c1 76784,C12(NC(c3c(C)cc(=N)[nH]c3)=O)COCCC1CN(C(c1c(Cl)n[nH]c1C)=O)C2 76785,c1(C(N(C)C)C2CC2)cn(CCC(N2CCCC2C(N)=O)=O)nn1 76786,N1(C(C(CC)N(CC)CC)=O)CC(NC(=O)CC(CC)C2CC2)C(C)C1 76787,N1(C(C(CCC)NC(=O)CCCNC(N)=O)=O)CCOC(C)(C)C1C 76788,n1(CC)ncc([N+](=O)[O-])c1C(=O)NC1CCCC(NC(c2csc(C)n2)=O)C1 76789,CC1(C)CN(C(C23CC(NC(=O)C=Cc4ccc[nH]4)(C2)C3)=O)C1C1CC1 76790,C(=O)(C1=NN(CC(C)C)C(=O)CC1)N1CC(N(C(C(CC=C)(C)N(C)C)=O)C)C1 76791,C12(C(N(CC(=O)OCC)C)=O)CC1CCN2C(=O)CC(C)C1CC1 76792,c1(C(=O)NC2CCC(NC(c3cc(C(C)=O)sc3)=O)C2)ccc2c(c1)ncn2C 76793,N1(C(C(C2CCC2)OCC)=O)CC2CCC1C2NC(c1nccnc1CC)=O 76794,c1(OC)ccnc(C(N2CC(NC(C3OCC4CCCC34)=O)C(SC)C2)=O)c1F 76795,C(C(C(F)(F)F)Nc1cccc(OCC(=O)OC(C)(C)C)n1)N(C)C 76796,c1(C(CO)N(C(=O)CC2(CN)CCOCC2)C)ccc(F)cc1 76797,c1(N2C(CC)CN(C(=O)Cc3cccc(SC)c3)CC2)ncc(C#N)cc1Cl 76798,C1(CNC(c2cnc(C(C)O)s2)=O)C2CN(C(=O)Cn3cc(C(N)=O)nn3)CC12 76799,c1(OC(C)C#N)cccc(CC(N2CCCCC2C2CCN(CC(N)=O)C2)=O)c1 76800,Cc1ccc2c(c1)CCN2C(c1ccc(NC(=O)Cc2nncn2C)cc1)=O 76801,c1(NCc2n(C(C)C)cnc2)ccc(F)c(C(=O)O)c1 76802,Cc1ncoc1C(=O)NCC1CCCC1NC(=O)C(C)c1ncco1 76803,C=CCCN=C(NCc1ccnn1C1CC1(F)F)NC1CCCC(NCC)C1 76804,Cc1ccc2cc(C(N3CCN(C(c4cnc(O)n(C)c4=O)=O)CC3C)=O)[nH]c2c1 76805,C1(C(=O)NCC)CN(C(=O)C(CC)NC(=O)Nc2nc[nH]n2)CCC1O 76806,C1(NC(C2(CNC(C(CC)C)=O)CC2)=O)CC(=O)N(CC(=O)NC)C1 76807,C1(CNC(CCNS(CC)(=O)=O)=O)CCCC2(CCN(C(=O)C(C)OC)CC2)O1 76808,C1(C(=O)NC2(C3CN(C(c4[nH]cc(C(C)=O)c4)=O)C3)CC2)CCCC(C)(C)CC1 76809,C1(C(=O)NCC(C)C(=O)N(C)C(c2ncccn2)C)C(C)(C)C1(C)C 76810,C1(C)CN(C(c2cc(C)sn2)=O)CCO1.CCCCCOCCN(CNC)C 76811,c1(CNC(C(COCC)NC(=O)C=CC(C)CC)=O)ccc(F)cc1F 76812,c1(OC)ccc(C(c2nn[nH]n2)N(C2(C#N)CCOC2)C2CC2)cc1 76813,c1(CC(C)C)cc(C(=O)NCc2ccc(C(=O)NC3CC(O)C3)cn2)n(C)n1 76814,C#Cc1cc(F)c(C(=O)NCC(C)N(C(c2cc(C)c(F)cn2)=O)CC)c(F)c1 76815,C=C(C)CC(C(=O)NCC(=O)N(C)CCN(C)CCOC)OCC 76816,c1(CNC(N2CC(N(C(=O)CC3(C)CCC3)C)C2)=O)cc(Cl)ccn1 76817,c1(C(C(=O)Nc2ccc(Cl)cc2F)N(C2CCOCC2)CC)ccc2occc2n1 76818,N1(C(CCCCN(C)C(c2cc(C#N)c[nH]2)=O)=O)CC2C(C1)C2(F)F 76819,C1(C(N2CC(C(C)NC(=O)COc3cccc(F)c3)C2)=O)CCc2nc[nH]c2C1 76820,c1(C(c2n(CCC)nnn2)NCCCN2CCCCC2)ccnc(C)c1 76821,C(Cc1cn[nH]c1)(C(=O)NCc1csc(C2CC2)n1)NC(C=C(CCC)C)=O 76822,C1(NC(COC)=O)CC(NC(=O)CCc2c(F)cccc2F)C12CCC2 76823,CC(C)(CC(F)F)C(=O)N1CC(CNC(C2CCC(O)C2)=O)C(C)(C)C1 76824,C1(CCC(=O)NCc2ncsn2)CCCCN1C(=O)CN1C(=O)CNC1=O 76825,Cc1noc(Cl)c1CC(=O)NC1CN(CCCNC(=O)CC2(CO)CC2)CCO1 76826,C1(OC)CN(C(c2nn(CC)nc2C)=O)CC1C(=O)NC12CC(F)(C1)C2 76827,C1(NC(C(C)C2CCC2)=O)CC2CCC(C1)N2C(=O)CCCN(C)C(C)C 76828,c1(OC(C)C(=O)NCC(O)CNC(=O)C=CC=C(Cl)Cl)cccc(N)c1 76829,C1(F)(CNC(CCOCC#C)=O)CCN(C(c2ccnnc2O)=O)C1 76830,c1(C(=O)NC(CNC(C2C(OC)C2)=O)C2CC2)ccc(C(N)=O)nc1 76831,C1(CC(N2CCN(C(c3csc(Cl)c3)=O)C(CO)C2)=O)CCC2(CCC2)O1 76832,C1(CC)CC(C(=O)NC2CCCC(CO)C2)CCN1C(=O)C(C(C)(C)C)OC 76833,c1(-c2nnc(N3CC(OC)C4(C3)CC4)n2C(C)C)oc2ccccc2c(=O)c1C 76834,N1(C(CC(C)NC(C2(C(N)=O)CCC2)=O)=O)CC2OC(=O)N(C)C2C1 76835,c1(C(=O)OCCNC(=O)OCC)cnc(O)c(F)c1 76836,c1(C(=O)NCC(C(=O)NCCCCCC=C)CC2CC2)ncc(F)cc1C 76837,c1(C(CC)Nc2cc(OC)ccc2OC)cc(C)cc(Br)c1OC 76838,CC1CCCN(C(c2ccc(CF)cc2)=O)C1CNC(C1CC2CC1C1CC21)=O 76839,N1(C(C(C)CC2CCCC2)=O)CCCCC1C1(NC(C2CCCSS2)=O)CC1 76840,C1(N(C(=O)CC2CC2(C)C)CC)CCN(C(=O)C(n2ccc(Br)n2)C)C1 76841,C(=O)(C1=C(CCOC)N(C(CC)CC)C(=S)NC1c1cc(OCC)cs1)OCC 76842,CC1CC2(C(=O)N(CC(C)N(C)C(c3csc(Br)c3)=O)C)CC12 76843,C(=O)(CC(C)(C)CN(C)C)NC1(C)CN(C(C2N(C(C)=O)CSC2)=O)C1 76844,C=C(I)CC(=O)NCC1(NC(=O)CN2CCCCC2)CC1 76845,C(=O)(C1=NOC(C)(C)C1)N1CCCC(NC(c2c(C)sc(C(F)(F)F)n2)=O)C1 76846,C1(C(=O)NC2C(C)CN(C(c3ccc(CN=[N+]=[N-])cc3)=O)C2)CCCCN1N=O 76847,c1(C(=O)NCCN(C(COCCC)=O)CCc2ccccc2)cccn(C)c1=O 76848,C1(C(=O)NCC=C(COC)C)(CNC(=O)CC(=O)NCC2(CF)CC2)CCCC1 76849,c1(CC)cc(C(=O)NCC(C)(C)OCCNC(=O)C(C)CC2CCCC2)c(C)o1 76850,C1(NC(C(=O)NC(C)C(CO)NC(=O)OC(C)(C)C)=O)Cc2ccccc2S1 76851,N1(C(C(C)=C(C)C)=O)C(C(=O)NCc2ccc(O)nc2)CCC1C(C)C 76852,N1(C(C2CCN(S(C)(=O)=O)C2)=O)CCOCC(C)(C(C2CC2)NC(=O)CSC)C1 76853,Cc1ccc(F)cc1C(=O)NCCC1(CNC(=O)C2CC2)CCCC1 76854,c1(C(=O)NC(C2CCOC2)C2CC2)cc(C2CC2)ncn1 76855,N1(C(C(COC)OC)=O)CC2(CC(NC(c3cnnc(C)c3C)=O)CO2)C1 76856,CC1CC=C(C(=O)NC(C(=O)NCCc2ncon2)c2cccs2)CC1 76857,C(=O)(CCC[N+](=O)[O-])N1CCCC(N2CCN(C(=O)Cc3cn[nH]c3)CC2)C1 76858,C1(CNC(CC(CN(C)C)O)=O)C2CCCC1N(C(c1csc3nnsc13)=O)C2 76859,C(=O)(CCCCN(C)C)N(CC(=O)N(C(C=C)C1CC1)C)CC 76860,C(=O)(C1=NNC(=O)CC1)NCC1C(NC(C(CCC)NC(C)=O)=O)COC1 76861,C(C(C)C(=O)N(C)CCOC1(COCCN(CCSC)CC)CCOC1)OC 76862,Cc1cccc(OC(C)C(=O)NCCCNC(C2(CC3CCC3)CCCC2)=O)c1 76863,C1(O)(C(C)NC(=O)CC2(O)CCOCC2)CCN(c2cc(C(F)F)ncn2)CC1 76864,CC1CN(C(=O)CC2(NC(c3ccc(F)s3)=O)CCCCC2)CC1F 76865,CC(O)C(C)(C)C(=O)N(C)CC1CN(C(c2ccc(CN(C)C)cc2)=O)CCO1 76866,c1(C(N2C3CN(C(CC=C=C)=O)C(C3)C2)=O)cc2c(s1)CCCC2 76867,N1(C(CC2CCC(C)CC2)=O)CC2(CCN(C(=O)C(C)C)CC2)C2COCC12 76868,C(C(=O)NOCC1CC1)N(C(=O)C=Cc1cc[nH]c1)CC#C 76869,c1(NC(C2C(C(=O)NC)C2)=O)cc(Br)cn2ccnc12 76870,N1(C(C)=O)CCCCC1C(=O)NCCCCC(C)NC(=O)Cc1ccc(F)cc1 76871,C(=O)(C1CCCc2cncn21)NC1CC(NC(Cc2ccc(C#N)cc2F)=O)C1 76872,c1(OCCNC(=O)Nc2cnn(C)c2CCC(F)(F)F)cccc(Cl)c1Cl 76873,c1(-c2cc(C(N(C3CN(C(Cc4c(C)cns4)=O)C3)C)=O)on2)ccccc1F 76874,C(=O)(C(C)C(O)CC)NCCOC(CNC(c1ccc(OC)nn1)=O)(C)C 76875,Cc1nc2ccncc2cc1C(=O)N(C1CN(S(=O)(=O)C2CCOCC2)C1)C 76876,c1(NCCCC(C)NC(COCC)=O)ncnc2c1cnn2C(=O)OCC 76877,c1(C(=O)NCC(CC=C)NC(C2CC(Cl)(Cl)C2)=O)cnn2cccnc12 76878,N1C(=NCc2ccccc2)N2CCC(C2)OCC1C.CC1CN(CC)CC(C)O1 76879,C1(NC(C(=C(C)C2CC2)F)=O)CC(C)N(C(=O)Cn2cncc2C)C1 76880,Cn1ncc2c(SCC(=O)NCc3cccc(Cl)c3)ncnc12 76881,c1(C(=O)NC2CC(NC(C3CCC(F)(F)C3)=O)C2)cc(Br)c(Br)s1 76882,C1(OC)CCCN(N(Cc2cccc(C)n2)CC(F)F)C1 76883,C(=O)(C1=CC(O)C(NC(C2(C(N)=O)CCC2)=O)C1)Nc1c(CC)noc1 76884,N1(C(CC(C)CNC(c2ccc3c(c2)CC3)=O)=O)CCC2(C=CCO2)C1 76885,C1(C2N(C(c3c(C)noc3)=O)CCC2)CCCN(C(=O)CC(=O)N(C)C)C1 76886,N1(C(c2c(CC)con2)=O)CC2CCC1C(CNC(C13CC(OC)C1C3)=O)C2 76887,C#Cc1ccc(C)c(NC(C2CCN(C(C3CC(C)(C)CCO3)=O)CC2O)=O)c1 76888,c1(C(N2CC3(CCCN3C(C3CC34CC(O)C4)=O)C2)=O)ccc2cnoc2c1 76889,c1(C(N(CC(C)N(C(c2c(CC)noc2)=O)C)C)=O)nc(C)c(C)nc1O 76890,N1(C(CNS(C)(=O)=O)=O)CC2CC1CN2C(=O)CSc1ccccc1 76891,N1(CCNC(CCCC)=O)CCC(NC(c2nccc(C)n2)=O)CC1 76892,C1(C(=O)OC)CN(C(=O)C(N2CCC(NC(=O)NC)CC2)=O)C(C)CO1 76893,c1(C(N2C(C(=O)NC(C)C(=O)NCC(C)C)(CC)CCC2)=O)cn(C)c(=O)cn1 76894,C=CCCCCCCC(=O)NC(C)(CNC(c1cc(COC)ncc1)=O)CO 76895,Cc1cc(C(N2CCC(c3ccccc3)(NC(=O)CO)CC2)=O)c(C)cc1Br 76896,C(=O)(C(O)CCCc1ccccc1)NC1C(C)CN(C(c2ccnnc2O)=O)C1 76897,c1(C(N2CC(CC)C(NC(c3scnc3Cl)=O)C2)=O)ccc2c(O)nncc2c1 76898,c1(CNC(C(C2CCN(C(c3c(C)snc3)=O)C2)F)=O)ccn(C)c(=O)c1 76899,C12CCC(O1)COCC1(CC1)NCC(F)CN2C.C(C)(C)(C)O.OC 76900,C1(O)(CN(C(c2cnc(C(C)C)[nH]2)=O)C)CCCN(C(C2CC23CC(O)C3)=O)C1 76901,C1(C(=O)NCCN(CCOC)C(c2ccc(C(F)F)o2)=O)CC2(C)CC1CO2 76902,CCCC(C(=O)NCCC1CN(C(c2nc(Cl)sc2Cl)=O)CCO1)NC(N)=O 76903,c1(C(N2CCCC(NC(c3nccc(C)c3)=O)C2C)=O)cnc2c(F)cccn12 76904,C=CCCC(C)(c1nnnn1C(C)(C)C)NC(C)CCO 76905,N1(C(C(C(C)C)n2cnnc2)=O)CC(N(C)C(c2ccc(F)cn2)=O)C(C)(C)C1 76906,N1(C(C(=O)NC)C)CC2C(NCc3noc(-c4ccccc4)c3Br)C2C1 76907,Cc1cc(Br)ccc1C(=O)NCCC1CN(C(=O)C(C)NC(N)=O)C1 76908,c1(C(=O)OC)csc(C2CCCN2S(=O)(=O)CC2CN(C)C2)n1 76909,C1(C(=O)NC2CC(OC)CN(C(=O)COCC3CC3)C2)CCC2(CC1)OCCO2 76910,C1(C(=O)NC23CC(C(=O)NCc4cncs4)(C2)C3)CCC=CCC1 76911,c1(C(=O)NCc2ccc(C(=O)OCC)cn2)c(C(F)(F)F)nn(C)c1C 76912,CCC(C)(COC)C(=O)NCC(C)N(C(=O)Cc1cccc(C(N)=O)c1)C 76913,c1(C2C(C(=O)NCC(C)(C)CNC(C3COCCOC3)=O)C2)cccc(Cl)c1 76914,C12(CNC(c3cnns3)=O)CC1CN(C(=O)C(C1CCCCCC1)O)C2 76915,c1(NC2CCN(C)C2)cc(NCc2cc[nH]n2)ncn1 76916,C(CCC(=O)NCC(F)CNC(=O)CNC(c1ccsc1)=O)N(C(C)=O)C 76917,c1(OC)c(CNC(CCC=C(C)C)c2nnnn2C)ccc2ccccc12 76918,C(=O)(CC1=NNC(=O)C1)N(CC(C)NC(C1(c2ccccc2)CC=CC1)=O)C 76919,c1(CC(N2C(CN(C)C(C3CCCC3F)=O)COCC2)=O)ccc(F)c(Cl)c1F 76920,C1(C(C)CC(=O)NCC(C)(C)C)CCCN(C(=O)OC(C)(C)C)C1 76921,C(C(=O)NCC(F)CNC(C1(CCF)CCC1)=O)(C(C)C)NC(=O)OCC 76922,C#CC1(C(=O)NC2(CCCCO)CC2)CN(C(=O)Cn2cnc(C(N)=O)n2)C1 76923,Cc1oc(C#N)cc1C(N1CCC(NC(c2ccn(C)c2)=O)C(CO)C1)=O 76924,[N-]=[N+]=NC1CC(C(=O)NC2CCCSC2)N(C(=O)Cc2ccccc2O)C1 76925,C(=O)(CC(C)CC(C)(C)C)N1C(CNC(CCC#CC)=O)CC(O)C1 76926,C(=O)(C1=CCCSC1)N1CCC(CN(C)C(C2CCN(C)S2(=O)=O)=O)CC1 76927,C1(OCC(=O)NCC(CC)N(C(=O)CC2CCN(C)CC2)C)CCN(C)CC1 76928,c1(OCC(=O)NCC2CCC(NC(C(C(C)C)O)=O)CC2)cccc(S(C)(=O)=O)c1 76929,N1(C(CCOCC#C)=O)CC2CC(C1)N(C(c1ccc(OC(C)C)nn1)=O)C2 76930,C(=O)(N=c1cc2n([nH]1)CCOC2)NC1(O)CC2N(C(=O)OC(C)(C)C)C(CC2)C1 76931,c1(NC(C2CC(C)CN2C(=O)CCc2cccc(O)c2)=O)nc(Cl)nc(Cl)n1 76932,Cn1ccc(S(=O)(=O)N2CCC(C(c3ccc(CNC=O)cc3)=O)CC2)c1 76933,C1(CC(=O)NC(c2cscn2)C)CC2(CC2)CN1C(c1cccc(F)c1N)=O 76934,c1(C(=O)NC2CCC(CNC(c3csnn3)=O)C2)c(F)ccc2n[nH]cc12 76935,CCCCCCOC(C)C(=O)NCCOC1CCN(C(=O)CSSC)C1 76936,c1(C(=O)NC2(CF)CCN(C(CCC(=O)OC)=O)C2)cc(C)cc(Br)c1F 76937,c1(NCC2(CC=C)CCCC2)ncccc1S(=O)(=O)NCCC1CCCC1O 76938,C(CC)(C(C)(F)F)NC(CN(C(=O)CN(C)C(C)C)CC)=O 76939,CC1=NOC(C(N2CC(NC(=O)C(C)COc3ccccc3)C2)=O)C1 76940,N1(C(C=CCOCCOC)=O)CC2CC2(CNC(C2CCOC2C2CC2)=O)C1 76941,C1(NC(CN2C(C)CCC2)=O)COCCC1NC(c1cc(CO)[nH]n1)=O 76942,Cc1c(C(=O)NCCNC(C23CC(C2)C3)=O)oc2c(F)cccc12 76943,C1(C(N2CC(NC(C=COCC)=O)CC3(C2)CCC3)=O)Nc2ccccc2C1(C)C 76944,c1(OCC(=O)NC(C(C)C)(C)CNC(C2(C#N)CCCO2)=O)ccc(F)cc1Cl 76945,c1(C(=O)NCC2N(C(CC3CC(=O)C3)=O)CCCC2)ccc(Br)c(F)c1 76946,c1(C(=O)NCC(CC(C)C)NC(CNS(CC)(=O)=O)=O)ccc(O)c2ccccc12 76947,N1(C(Cc2nc(NC(=O)Nc3ccnc(O)c3)sc2)=O)CCCC(F)(CO)C1 76948,C1(CCC)CN(C(c2c(N)sc(C)c2C)=O)CCN1C(c1cnn2c1OCC2)=O 76949,N1(C(C(=Cc2cccs2)C)=O)CCC(C2CC2)C1CNC(c1ccoc1C)=O 76950,C1(C(N2CC3C(CO)C3C2)=O)C(O)CCN1C(c1cccnn1)=O 76951,Cc1nc2nccc(N(C(C)CNC(c3cc(F)cnc3O)=O)C)n2n1 76952,c1(C(=O)NC2C3N(C(C(C)C#N)=O)C(CC3)C2)nnn2c1C(=O)NCC2 76953,CCC(C#N)C(=O)N(CC(C)C(=O)NC(C1CCCCC1)C)C 76954,n1(CC)cc(C#N)c(=NC(=O)c2cc3c(cc2SCC(=O)OC)OCCO3)[nH]1 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77235,c1(CCC(=O)NCC2C(NC(C3CC(OC(F)F)C3)=O)COC2)nnc(S)nc1O 77236,N1(C(CNC(C(CC)C)=O)=O)CCN(C(C2(C(C)C)COC2)=O)CC1CC(F)F 77237,c1(C(=O)NCC2N(C(C(COCC)C)=O)CC=C2)cnn2ccsc12 77238,N1(C(C2N(C)C(=O)CC2)=O)CCCN(C(=O)CCCCC#N)CC1c1ccccc1 77239,c1(C(=O)NCC(C(C)C)NC(c2cccc3nn[nH]c23)=O)ccnc2[nH]ncc12 77240,C1(C(=O)NOCC2CCCC2)(CC=C)CCCN1C(c1ncccc1O)=O 77241,C(=O)(C(C)(C)CCCC=C)NC(C(N1C(C#C)CC1)=O)COC 77242,C1(CCOC)(CNC(c2ccns2)=O)CCN(C(c2csc(C(C)OC)n2)=O)C1 77243,Cc1c(F)ccc(C(=O)NC2(CNC(C3CCCCO3)=O)CCOC2)c1O 77244,CCC(C)CCCC(=O)N1CC(F)CC1CC(N1CC(CO)C2(CC2)C1)=O 77245,N1(C(c2c(COC)noc2)=O)CCC(N=c2cc[nH]cc2C#N)CC1C 77246,N1(C(C2(CC=C)CC2)=O)CC2(C1)CN(C(C1Cc3ccccc3O1)=O)CC2CO 77247,c1(NCC(=O)NC2CN(C(C=C(C)C(C)C)=O)C2)cccc(C#N)c1 77248,C1(CC(=O)N(C(CNC(C2COC(=O)N2C)=O)C2CC2)C)CCCCC1(C)C 77249,C1(CNC(C2CN(CCOC)C(=O)C2)=O)(CO)CCN(C(=O)CSC)CC1 77250,C=CC(C)C(C)C(=O)N1CC(OCCNC(c2ccc(N(C)CCC)nc2)=O)C1 77251,C1(C(N2CCC(N(C(=O)CCC3CCCCC3)CCO)C2)=O)COCCC1CO 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77286,c1(OC(C(CC)(Cc2ccc(OC)cc2)CC)=O)ccc2c(=O)[nH]ccc2c1 77287,c1(C(N2CC(NC(C3(COC)CCCC3)=O)C(F)C2)=O)cc(C)nnc1C 77288,C1(C(=O)NCC2CCN(C)C2)(OC)CCN(C(=O)Cc2cc(C3CC3)no2)CC1 77289,c1(C(=O)NC2C(OC)CN(C(=O)C(C)CSC)C2)cc(C)c(OC)c(C)c1 77290,CCCC(C)(C)C(=O)NC(c1ccccc1)CNC(=O)C(C)(CC)CC 77291,Cc1ncnc(C)c1C(=O)NCC(C)(C)CNC(C1CCOC1(C)C)=O 77292,N1(C(COCCC#C)=O)CC(C(=O)NCC(C)C(C)O)C(CC)C1 77293,c1(C(N2C(C(N(C)C)=O)C=CC2)=O)cc2cc(Br)ccc2o1 77294,C1(NC(C2N(C(C)=O)CCC2)=O)CCN(C(=O)CSc2ccccc2)C1(C)C 77295,N1(C(c2c(OC)n[nH]c2)=O)CC2(CC(CC(N3CC4CCC4(C)C3)=O)C2)C1 77296,O(C=CC(=O)N(C)CC1(NC(=O)Cc2ccco2)CC1)CC 77297,N1(C(C2NC(=O)OC2)=O)CC2CCCC(NC(c3cc4ncccc4s3)=O)C2C1 77298,c1(-n2c(-c3ccc(C(F)F)cc3)nc(C)n2)ccc(-n2cnnc2)cc1[N+](=O)[O-] 77299,c1(C(=O)NC(C)CN(C(=O)C(Cc2ccccc2)N(C)C)C)c(O)cncc1F 77300,c1(C(=O)NC2(CNC(C(CC)NC(N)=O)=O)CC2)ccn(C)c(=O)c1 77301,c1(OC)ccccc1C(C(=O)OC)N(C1CCN(C(c2cnn(CC)c2)=O)C1)C 77302,N1(C(C(C2CCN(C(C3COCCC3C)=O)CC2)C)=O)CC(N(C)C)CC1CO 77303,N1(C(C(C(C)(C)C)OC)=O)CCCC2(C1)CN(C(c1cc(C)c(C#N)cn1)=O)C2 77304,Cc1c(C)n(C)c2ccc(C(=O)NC3CCOCC3NC(C3CC(O)C3)=O)cc12 77305,C=CC1OCCCC1C(N1CCC(OCCNC(c2nn(C)c(C)c2Cl)=O)C1)=O 77306,c1(OCC(=O)NC(C)C(C)NC(=O)CN2CCNC2=O)ccccc1Cl 77307,N1(C(CC(O)C(F)(F)F)=O)CCc2sc(-c3cnn(CC(F)(F)F)c3)cc2C1 77308,C1(N(C(C(C)NC(CC)=O)=O)C)CCCN(C(c2cnn(C)c2COC)=O)C1 77309,C1(NC(c2ccc(C)o2)=O)(CNC(C2CCOCC2)=O)CC(F)(F)C1 77310,C1(CC)CN(C(c2ccc(Cl)nc2)=O)CCN1C(=O)CCc1cccc(OC)n1 77311,c1(CCCC)ccc(CC(=O)NC2CC2CNC(=O)C(C)OCC(C)C)cc1 77312,C1(C)(CC)CCC(C(=O)NCC(C(=O)NCCCc2cccnc2)N(C)C)O1 77313,c1(NC(C2(C)CN(C(=O)NCC(=O)OCC)C2)=O)cc(F)cc(F)c1C#N 77314,C=CCC(C)C(C)(c1nnnn1CCCC)NCC1CCC(F)(F)C1 77315,CC(C)(C)C(CNC(=O)Cn1ncnn1)C(=O)NC(CCO)C(C)(C)C 77316,N1(C(c2c(C)cccc2F)=O)CCN(C(C2CCCCNC2=O)=O)CC12CCC2 77317,C(=O)(CC(CC1CCCCC1)NC(=O)Nc1ccccc1)OC 77318,C1(F)(C(N2CC(OCCOC)C2)=O)CCCN(C(=O)CC2CCCSC2)C1 77319,Cc1cc2c(C(=O)NCC3(C)CCCN3C(=O)Cc3cnc[nH]3)nccn2n1 77320,N1(C(C(CCC)C(C)C)=O)CCN(C(=O)CC2CCCCC2(F)F)CC(C)(C)C1 77321,S(=O)(=O)(c1cccc(N2CCOC3(CCC3)CC2)n1)NC1CC(C)SC1 77322,N1(C(c2cncnc2)C(=O)NCC=C)CCc2cnn(-c3ccccc3)c2C1 77323,N1(C(C(CCC)C)C(=O)NC2COC2)CCc2c(CCC)cccc2C1 77324,c1(C(=O)NC(C)CCO)cccn1Cc1ccncc1 77325,C1(C(=O)NCC2CN(C(CCN(C(C)=O)C)=O)C2)CCCC(C(F)(F)F)O1 77326,C(=O)(CCC(C)OCC)NC(C1N(C(C(C=C)O)=O)CCC1)(C)C 77327,C12(C(NOCCNC(C)=O)=O)COC(CN1C(=O)COCCCOC1CCOC1)C2 77328,N1(C(CCC)=O)CCC(C(=O)NC2CC(C)(NC(C3CCCN3CC)=O)C2)CC1 77329,C#CCC(CC(=O)NC1(C(O)COC)CC1)NC(C1(CO)CCOC1)=O 77330,c1(C(C)=O)nc(C(=O)NC2CC2NC(c2cnn(-c3ccccc3)n2)=O)cs1 77331,c1(C(N2CCC(Cc3ccc(NC(C)=O)nc3)C2)=O)ccc(C#N)c(Cl)c1 77332,N1(C(c2cnc(CCC)s2)C(=O)NCCCSC)CCC(C(N)=O)C(C)(C)C1 77333,CC#CCCC(=O)NC1CC(C)(NC(c2cccc(-c3cnn(C)c3)c2)=O)C1 77334,c1(OC)cc(C(=O)NCC2CCC2NC(=O)CN2CC(C)C2)cnc1OC 77335,C12(NC(c3ccc(CCC)[nH]3)=O)CC1CN(C(=O)C(CC)n1cccn1)C2 77336,C1(CNC(c2c(OC)cccn2)c2nnnn2C2CCC2)CC2CCC(C1)O2 77337,c1(C(=O)NC(CC)CN(C)C(C2(C(N)=O)CC2)=O)cn(C)c(=O)c2cncn12 77338,c1(OC)ncc(C)cc1C(=O)NCC1(C)CCCN1C(c1ccn(C)c1)=O 77339,C1(CNC(COCC#C)=O)CCC(NC(=O)C(N2CCNC2=O)C)C1 77340,c1(C(=O)NC2(CNC(c3onc(OC)c3Br)=O)CCC2)ccc2c(c1)CCC2 77341,N1(C(COCC)=O)CC2COCC(C1)C2NC(=O)CCC1CCC(=O)N1 77342,c1(OC)ccc(CC(=O)NC2(C)CCN(C(=O)CSc3cccc[n+]3[O-])C2)nc1 77343,C1(CC(=O)NCCCOCCOCCNC(C(C)C)=O)CC=CCC1 77344,N1(C(C2(C)CC2)=O)CC2(CCN(C(C3C4CCC3(c3ccc(F)cc3)C4)=O)C2)C1 77345,C=Cc1ccc(C(N2CCC2C(=O)Nc2ccc(C(F)(F)F)nc2)=O)cc1 77346,c1(CC)ccc(C)cc1C(=O)NCC(CNC(c1ccc(C)o1)=O)S(C)(=O)=O 77347,c1(C(N(CC(=O)NC2CCC(C#N)C2)CC2CC2)=O)coc2c1COC2 77348,c1(NC(C(C)N(C(=O)COCCCN=[N+]=[N-])C2CC2)=O)cncc(Cl)c1 77349,C(=O)(C(F)CC(C)(C)NC(=O)Cc1ccc(F)cc1)N(C1C(C)C1)C 77350,c1(NC(C2CCN(Cc3c(Br)ccnc3Cl)C2)=O)cccc2nsnc12 77351,N1(C(C(C)CCN(C)C)=O)CCC2(CCC(NC(=O)Cc3nccn3C)CC2)C1 77352,c1(C(C(=O)NC(C)C)N(C(CC)CC)C(C)CC)cc2c(cc1OC)CCC2 77353,C1(NC(Cc2n(C)ccc2)=O)CCN(C(=O)CCc2ncco2)CC12CCC2 77354,N1(C(=O)Nc2ccccc2Oc2ccc3c(c2)CCO3)CCN2C(=O)OCC2C1 77355,C#CCC(CC#C)C(=O)N(C1CCN(C(=O)CC2(CO)CC2)CC1)CC 77356,C1(C(=O)NCCn2cc(C3(C)CC(O)CN3C)nn2)(OC)CCC(C)(C)C1 77357,N#Cc1c[nH]cnc1=NC1COC2(CCN(C(=O)C3=CCCCO3)CC2)C1 77358,C1(c2n(Cc3nnn(C)n3)nnn2)(Nc2nn(C)cc2Cl)CC2COCC2C1 77359,c1(NC(c2c(C)nc(C)o2)=O)cnc2c(c1)CN(C(=O)CC#N)CC2 77360,C1(C(=O)NCC2N(C(c3c(C)con3)=O)CC3(CC3)C2)CC=C(C(C)C)CC1 77361,C12(NC(c3c(OC)c(=O)cco3)=O)CCCC1CN(C(c1cc(=O)cc[nH]1)=O)C2 77362,CCC(C)C(=O)C(=O)N1CCC(F)(C(=O)N(C)Cc2ccncc2C)CC1 77363,N1(C(C2(Cl)C(C(C)=O)C2)=O)CCOC(c2cn(-c3cccc(C)n3)nn2)C1 77364,C12(NC(c3c(=N)[nH]cnc3)=O)CCN(C(=O)CCOC3CCC3)CC1C2 77365,C1(CC(=O)N(CCC(=O)NC(CN(C)C)CC)CC#C)CC(O)C1(C)C 77366,C1(C)(C(=O)OC)CN(C(c2cc(CNC(=O)CC3CC(F)(F)C3)[nH]n2)=O)C1 77367,CC(C)C(C)CC(=O)N(CC(O)CN(C(=O)Cc1nncs1)C)C 77368,O=S1(=O)CC2CN(Cc3cccc(OC(F)(F)C(F)F)c3)CC2(Cc2ccco2)C1 77369,c1(CS(=O)(=O)C(N2CCN(C(F)(F)CF)CC2)=O)csc2cc(Cl)ccc12 77370,CCCC(C(=O)N(CC(C)(C)NC(C1CC(SC)C1)=O)C)OCC 77371,c1(NC(=O)NCCc2ccc(CC)cc2)ccc(Br)c(Br)c1 77372,N1(C(CN2CCC(C)C2)=O)CCC(CC(=O)NCC2(F)CCCCC2)CC1 77373,c1(C(=O)OC)cccc(C(N2CC3CC2C3C(=O)NCc2ccncc2F)=O)n1 77374,c1(CCC(N2CCC(NC(c3cccc(C)c3)=O)C2)=O)c(F)cccc1Cl 77375,N1(C(CCC=C(C)C)=O)CCCC(NC(=O)COc2cc(C)on2)C1C 77376,CS(=O)(=O)c1cnc(C2CCN(C(=O)COc3ccsc3)CC2)nc1 77377,CC1CCC(C)C1NC(=O)CC1CCCC1NC(=O)Cc1cnns1 77378,c1(C(=O)NC2CC(F)(CNC(C=C(C)C)=O)C2)cc2scc(C)c2[nH]1 77379,c1(NC2CC(C)(C)OC2)cc(Br)ccc1S(=O)(=O)N1CCC(C2CC2(F)F)CC1 77380,C(=O)(CC(C)(C)C(=O)OC)NC(CCC#C)C(=O)N1CCC12CCCC2 77381,C(=O)(CC(COC)NC(C1(C)CNC(=O)N1)=O)NCc1ncc(CC)[nH]1 77382,C(=O)(C(C)CC(C)(C)C)NC1(CC(N2CCC(COCC)CC2)=O)CCOC1 77383,c1(C(=O)NCC(C2CC2)NC(=O)C2=CCS(=O)(=O)C2)cnc2ccc(F)cn12 77384,C1(C(=O)NC2CCCC2CNC(=O)CCc2ccncc2)(COC)CCCC1 77385,Cc1onc(CC(=O)NC(c2ccc(C(C)C)cc2)C)c1-c1nn[nH]n1 77386,c1(C(=O)NCC2N(C(C#CC(C)C)=O)CCC2)nccc2c(Cl)cccc12 77387,c1(C(=O)NC(C(C)NC(c2cccc(CO)c2)=O)C)ccc(O)c(N)n1 77388,n1(CC(=O)NC2CN(C(C(C=CC)O)=O)CC(C)(C)C2)c(=O)oc2ccccc12 77389,N12CC(O)C(O)C(O)C1C2.c1(C(=O)OCC)ccc(O)nc1CN 77390,c1(C(N2CCC(F)(CNC(C3C(C)C3)=O)C2)=O)cc(-c2ccccn2)cc(F)c1 77391,C(=O)(C(c1cccs1)N(C)C(C)C1CC1)NCCSC 77392,C1(C(=O)NCCc2c(CNC(C(C=CC)O)=O)nco2)CCCC(CF)C1 77393,C(CNC(=O)C(C)C(F)(F)F)(CC(F)(F)F)NC(c1cccc(C(C)C)c1)=O 77394,Cc1ccc(Br)c(C(=O)NC2(C)CCN(C(c3c(C)cccc3O)=O)C2)c1 77395,c1(NC(C(C2(C)CC2)NC(CC2C(C)(C)C2)=O)=O)cnc2ccnn2c1 77396,C1(N(C(c2c(COC)nn[nH]2)=O)C)CN(C(=O)C(C)N(C2CC2)CC)CCC1O 77397,c1(C(=O)NC2C(C(N(CC(F)(F)F)C)=O)C2)ccc2cnccc2n1 77398,C(=O)(C(F)CCC(C)(C)C)NC(CN(C)C)C(N1CCC(CO)C(C)(C)C1)=O 77399,S(=O)(=O)(c1nc(N2CC(CO)C(C3CC3)C2)ccc1Br)N(CCF)CC 77400,CC(CC(C)(C)O)NC(=O)C(Cc1ccccc1Br)NC(=O)C=Cc1cscn1 77401,C(CCCCC(=O)NC1CCCCCC1C(=O)NCCC(C(C)C)OC)OCC 77402,Cc1c(C(=O)N(CCCNC(C2CC(C(C)(C)C)C2)=O)C(C)C)nnn1C(C)C 77403,CCC(CC(F)F)C(=O)NCC1(F)CN(C(C2(C3CCCCC3)CC2)=O)C1 77404,N1(C(C2C(C)(CC)C2)=O)Cc2nccn2CC(NC(=O)C(c2cnn(C)c2)C)C1 77405,Cc1cc(C(=O)NCCN(C(=O)C(F)F)C2CC2)n2ncnc2n1 77406,C#Cc1ccc(C(=O)N(CCCNC(c2cc(C)n(CCO)n2)=O)CC)c(C)c1 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77603,C(=O)(C1CCCn2c(Br)cnc21)NC1CC(NC(c2ccc(C#N)[nH]2)=O)C1 77604,Cc1cc(N2CCN(C(C3CCCC4(CC4)C3)=O)CCC2C)n2ncc(C)c2n1 77605,C1(O)(COC)CCN(C(C2CC(CNC(=O)C(C)(F)c3ccon3)C2)=O)C1 77606,N1(C(C2C(CNC(CCOC(C)=O)=O)CC2)=O)C2CCC1CC(C(N)=O)C2 77607,C1(C(=O)NC(c2ccnn2C)C)CCCCCN1C(C1C=CCS1)=O 77608,c1(CC(=O)N(CCCNC(c2nc(C)sc2C)=O)C(C)C)cc(F)ccc1Cl 77609,C(=O)(C(O)Cc1cnc[nH]1)NC(C1CCCCC1)(CNC(C(C)C1CC1)=O)C 77610,c1(C(N2C3CC(CN(C(Cc4cnn(C)n4)=O)C3)C2)=O)ccc([N+](=O)[O-])cc1F 77611,O=C(CC(=O)c1ccccc1)NC1CC1NC(=O)C(c1ccccc1)O 77612,C1(N(C(C2C(C)OC(=O)N2)=O)C)CCCN(C(=O)CC2CCCCC2(C)C)CC1 77613,C1(OC)CCCN(C(C2CC(O)CN2C(c2ncncc2N)=O)=O)CC1 77614,c1(SC)nc(O)nc(C)c1C(=O)NC1CCCCC1NC(=O)C1=CCCCC1C 77615,C1(CCNC(C(C)(C)SC)=O)CC2CCC(C1)N2C(=O)CC1CCCS1(=O)=O 77616,Cc1ccc(C(=O)NC(C)(C)CC2CCN(C(C3(O)CC3(C)C)=O)CC2)nc1 77617,n1(CC)cnc2nc(=NCC3CCCC(CO)C3)[nH]c(NCC3CCCC3)c12 77618,N1(C(C2NC3CCC2C3)=O)CCOC(Cn2cc(-c3ccoc3)cn2)C1 77619,C1(NC(c2ccc(C(C)=O)cn2)=O)CCC(C)N(C(C2CCOC2)=O)C1 77620,C1(C(=O)NCCn2ncc(C)c2)CCCN(C(c2scnc2C(C)C)=O)C1 77621,N1(C(C(=O)Nc2cc(OC(C)C)cc(OC)c2)=O)CC2CCCN2CC1CO 77622,C1(C(N2CCC(CF)(NC(c3cnco3)=O)C2)=O)(CC)CCNC1=O 77623,c1(SCCN(C(c2nc(C)sc2)=O)C)cccc(NC(=O)C(C)C2CC2)c1 77624,c1(C(C)OC(CCC(C)NC(C(C)C2CC2)=O)=O)cccc([N+](=O)[O-])c1 77625,c1(OC(C(=O)NC(c2c(C)noc2C)C(F)(F)F)CN(C)C)cc(Cl)cc(Cl)c1 77626,N1(C(CSCC#C)=O)CCN(C(=O)C=C2CCC(C)CC2)C(CC(F)F)C1 77627,c1(CNC(C(CO)NC(CC2CCC(=O)NC2)=O)=O)cc(O)ccc1F 77628,CCCC(C(O)C(=O)N(CCOCCO)CC)NC(c1ccn(C(C)C)n1)=O 77629,C#CCC(C(=O)NN1CCCC1C(=O)NCC(O)C(N)=O)C1CC1 77630,c1(CNC2C(C(=O)NCCC#N)CCCC2)cc(O)c(O)c(O)c1 77631,C1(NC(c2scc(COC)c2)=O)C2CCN(C(c3c(CO)n[nH]c3C)=O)CCC12 77632,C12(CCNC(CCCC=C)=O)CCC(CC1)N(C(c1ncn3c1CCC3)=O)C2 77633,c1(C(=O)NCC2C=CCN2C(=O)C=CBr)c[nH]c2ccc([N+](=O)[O-])cc12 77634,N1(C(c2c(C)nc3sccn32)=O)CCCC2(CCCN2C(c2ccnn2C)=O)C1 77635,C1(NC(CCCCOC)=O)CC2CCC1N2C(=O)C(C)Cc1cccc(Cl)c1 77636,C#CC1(OCC(=O)N(C2CCN(C(C3(C(C)(C)OC)CC3)=O)C2)C)COC1 77637,C(N=c1cccc(S(=O)(=O)NC2CCC=C2Br)[nH]1)C1CC(C)(C)OC1 77638,C=CC1(C(=O)NOCC2CCC2)CCN(C(=O)CC2CCCNC2=O)C1 77639,c1(CC(=O)NCC2CCN2C(c2cc(C(F)F)no2)=O)ccccc1Br 77640,c1(C(=O)NC2CCCCN(C(CCC=C)=O)C2)cc(S(N)(=O)=O)c(F)cc1OC 77641,C(=O)(C1=CS(=O)CCC1)NC1CC(N(C)C(C2CC2c2ccccc2)=O)C1 77642,c1(C(N2CC(NC(=O)Cc3cccnc3Cl)CC(C)C2)=O)c[nH]c2ccccc12 77643,N1(C(C2(COC)CCC2)=O)CCN(c2ccc(C(=O)NC3CCSC3)cn2)CC1 77644,c1(CC)ccc(F)cc1F.c12c(cnn1C(C)(C)C)NC1(CCO)CCCC1C2 77645,N1(C(c2c(CNC(CCc3ncn(C)c3)=O)c[nH]n2)=O)CCCC(N=[N+]=[N-])CC1 77646,CC1CN(C(C2C3CCC(C3)C2NCc2ccc(F)cc2)=O)C(C)(C)C1 77647,C1(C(=O)NCCN(CC(C)O)C(c2ccoc2Cl)=O)CCn2c(O)nnc2C1 77648,C1(NC(CC2(N(C)C)CC2)=O)C=CC(CNC(=O)CC2CC(F)C2)C1 77649,C1(CNC(c2n(CC)cnn2)=O)CCCCN1C(C1OCCOC1C(F)(F)F)=O 77650,c1(C(C)NC(=O)OC(C)(C)C)ccc(OC(F)F)nc1.C12CC(C)(C1)NC2=O 77651,C(=O)(C(C)N=c1[nH]c2ccccc2s1)NC1CC(CNC(CCCCC#C)=O)C1 77652,CC(C)(C)CCNC(N1C(C(=O)Nn2cc(C#N)cn2)COCC1)=O.C1CC1 77653,Cc1cc(C(N2CCC3(CC3NC(C3NC(=O)OC3C)=O)C2)=O)ccc1F 77654,CN1CC(CC(N2CC(F)(CNC(c3csc(C(F)(F)F)n3)=O)C2)=O)CC1=O 77655,C1(CC(=O)NCC(CC)NC(=O)CCN2CCC(O)CC2)Cc2ccccc2O1 77656,N(C1CCC(NC(C2(CO)CCCC2)=O)c2ccccc21)C(c1c(C)[nH]cc1)=O 77657,C1(NC(COCCSC)=O)CCC2CCN(C(c3cncc(Cl)c3)=O)C1C2 77658,c1(C(N2CCC(NC(c3ccc(OC)s3)=O)(CF)C2)=O)cc2sc(C)nc2[nH]1 77659,C1(C(N(CCCNC(CNS(CC)(=O)=O)=O)C)=O)CC(F)(F)C1(F)F 77660,Cc1ccc(OCC(=O)N(CCNC(C2(C(C)C)CNC(=O)C2)=O)C2CC2)cc1 77661,C(N=c1[nH]cc(Br)c2ccc(Br)cc12)C1C(O)COC1 77662,C1(CNC(C(N2CCC(O)CC2)C)=O)CCCCC1NC(=O)C(O)C1CCC1 77663,Cc1cc2ccc(C(N3CCCC3C3(NC(=O)C4CC4)CC3)=O)cn2c1 77664,N1(C(CCS(C)(=O)=O)=O)CC(C)(CNC(c2csc(C3CC3)n2)=O)CC1(C)C 77665,N1(C(=O)OC)CCCC(C#N)(NC(c2ccc(C(=O)OC(C)(C)C)cc2)C)C1 77666,C(=O)(C#CC1(C)CC1)NC(CC)CNC(=O)CCC1CC1(Cl)Cl 77667,CCCC(O)CC(=O)NC1CC2CC1N(C(=O)CC(COC)COC)C2 77668,C12(C(=O)NCc3noc(Cc4ccccc4)n3)CCN(C(=O)C(O)CCl)CC1C2 77669,CC1CN(C(=O)CS(N)(=O)=O)CC(C)CN1C(c1nccc(Cl)c1O)=O 77670,c1(C(=O)NCC23CC(NC(C#CC(=O)N(C)C)=O)(C2)C3)nnc2ccccn12 77671,Cn1nc2c(c1C(N1CC(NC(C3CCOC3)=O)C(C(F)(F)F)C1)=O)CCC2 77672,C1(N(C(Cn2c(C)ncc2)=O)C)CN(C(C2CC(F)(CO)C2)=O)CC1O 77673,c1(CC)cc(Cl)ccc1C(=O)NC1CCC1CNC(c1ccccc1C)=O 77674,C1(NC(c2cc(C)oc2C)=O)CC2(C1)CC(NC(=O)Cc1c(F)cncc1Cl)C2 77675,C1(N(C(C2CC2C#N)=O)CC)CCC(NC(C2CC(C)=NO2)=O)CC1 77676,c1(NCc2nn(CC)nc2C)cc2c(I)cnn2cn1 77677,C(=O)(C(F)(F)CC(C)C)NC(CN(C(c1cnc2ccnn2c1)=O)CC)C 77678,O=C(CCC(F)(F)F)NCC1C(O)C(O)CN1C(=O)C(O)CN1CCCC1 77679,N1(C(c2cccc(C)n2)=O)CCC(C)C(N(C)C(C2CCCNS2(=O)=O)=O)C1 77680,N#CC1(C(N2CC3CC3(CNC(=O)CCc3cnc(O)[nH]3)C2)=O)CC12CCC2 77681,c1(C(=O)OC)cc(C(=O)N(C)CCN(C(=O)Cc2nccn2C)C(C)C)ns1 77682,c1(NC(C)=O)ccc(F)c(C(N2CCC(N(C(=O)CC3CC3(C)C)C)C2)=O)c1 77683,CC1=C(CNC(=O)C(C2CCN(C(=O)CC3CCC(=O)C3)CC2)C)CCC1 77684,c1(C(=O)NC(C2N(C(c3cc(C)sn3)=O)CCCC2)C)c(N)c(F)cc(F)c1F 77685,c1(C(=O)OC)cc(C(N2CCCC(C(C)(C)C)C2)C(=O)NCCCF)c(C)s1 77686,C=CC(CC)CC(=O)N1CCOCC1CN(C)C(c1cn(C(F)F)cn1)=O 77687,CC1(CNC(=O)CC2CC(O)CN2C(=O)COC2CC=CC2)CCCCCC1 77688,C1(N(C(c2sc(CC)c(C)c2)=O)C)CN(C(C23CCC(C2)C3)=O)CC12CC2 77689,c1(C(C)N(CCNC(=O)N(C)C)Cc2ccnc(Cl)c2)cccc(F)c1 77690,CC(C)C(O)CCNC(=O)C(CCOCCO)NC(c1cc(O)nn1C)=O 77691,c1(C(=O)OC)c(C)cc(C)nc1N1CCC(C)(NC(C2(C3CCOCC3)CC2)=O)C1 77692,C1(CC(=O)N(C)CC2CCN(C(=O)CS(N)(=O)=O)C2)CCC2(CCC2)O1 77693,CC1CC(NC(c2ccco2)=O)CN1C(C1CCCC(O)C1)=O 77694,c1(OC)ccc(CCC(=O)N2CC(NC(c3c(N)cnn3C)=O)C2)cc1F 77695,C1(NC(c2cc(CC)[nH]n2)=O)CCN(C(c2nc(-c3cccs3)no2)C)CC1 77696,c1(CCC(=O)NC2C(CN(C)C)CC2)csc(CSc2ncc[nH]2)n1 77697,Cc1cc(C)c(C)c(C(=O)NCC2(O)CN(C(c3coc(CO)c3)=O)C2)c1C 77698,c1(OC(C(=O)NCCCC(C)NC(C2(C=C)CCC2)=O)C)cccc(C)c1C 77699,C1(C(=O)NC(C)CN(C(=O)CNC(c2cccs2)=O)C)CC12CCC2 77700,C(=O)(CN=c1cc[nH]cc1)N1CC2C(CNC(=O)C(F)=C3CCC3)(C2)C1 77701,S(=O)(=O)(c1ccc(Br)cc1NCCc1cccnc1)N1CC(CCC)OCC1 77702,N1(C(C(C)Cc2ccc(F)cc2)=O)CC2CC(NC(=O)C3CC3)CC1C2 77703,N1(C(COCCC=C)=O)Cc2ccccc2C(CNC(C2(F)CC=CCC2)=O)C1 77704,c1(CC)cc(C(=O)NCCCCC(=O)NC(c2ncn(C)n2)C)c(C)o1 77705,C1(C(N2CCC(C(=O)NCC3CC(OCC)C3)C2)=O)CCCC(C#N)C1 77706,C(=O)(C1=CCC2CCC1N2C(C1(C)CSC1)=O)N(C)CC1CCCCO1 77707,CC(=O)CCC(=O)NCC(C(=O)NCC12CC(F)(C1)C2)N(C)C 77708,C(CC(C(=O)N(C(C)C(C)SC)C)NC(C1(CCC=C)CC1)=O)SC 77709,C1(C)(CNC(c2cnn(CC)c2C)=O)CCCN(C(c2c(C#N)cnn2C)=O)C1 77710,Cn1nnc(CNC(=O)C(C)(C)C#N)c1C(N1CC(CO)C1(C)C)=O 77711,N1(C(CSc2n(C)cnn2)=O)CCOC2(CCC(NC(=O)C=CCO)CC2)C1 77712,c1(C(N(C2CCCCC2)CCNC(C(CCCC)O)=O)=O)nn(C)c(=O)cc1C 77713,c1(CNC(=O)CCC2CC2)csc(C)n1.C1(N(CCOCCO)C=O)CC1 77714,N1(CCC#C)CCC(C(=O)NC2CCCC(CNC(=O)C(COC)CC)C2)CC1 77715,CCC(C(=O)NC(C1CCCN1C(=O)Cc1ccc(C)o1)C)OC 77716,c1(NC)ccc(C(N2CCCC2C(C)NC(=O)C(C)SC)=O)cc1 77717,c1(-c2nnc(N3CCCC(OCC)C3)n2CC2CCCO2)cc(Br)cc(F)c1F 77718,CC1CN(C(c2c(Cl)ncn2C)C(=O)NCCC2(C)CC2)CCN(C)C1 77719,NC(=O)CCC(=O)NC1CCCC1NC(c1ccc(Br)o1)=O 77720,C1(C(=O)NC2(CSC)CCC2)CCCCN1C(=O)Cn1cccc1 77721,C12SC3C=CC1CC3CN(C(=O)OC(C)(C)C)CC(F)CCCOC2=O 77722,C1(CNC(C2CCN(CCC#C)CC2)=O)CC2CCC1N(C(=O)C(C)C1CC1)C2 77723,N1(C(CCCCCNC(c2ccc(C(N)=O)o2)=O)=O)Cc2ccncc2C1 77724,c1(NC(C(N2CCC3(C=CCO3)C2)C)=O)nc2ccc(F)cc2s1 77725,N#Cc1ccncc1NC(C1CC=CC(n2cc(CC(=O)O)nn2)C1)C1CC1 77726,c1(C(N(C2C(C)CCN(C(c3cc(C)[nH]n3)=O)C2)C)=O)cnc(O)c([N+](=O)[O-])c1 77727,c1(CC(N2CC(N(C(=O)C(O)Cn3cncn3)C(C)C3CC3)C2)=O)ccccc1Br 77728,c1(CC(=O)N(C(c2cc(C)nc(N(C)C)n2)=O)C(C)C)ccccc1S(C)=O 77729,C(=O)(CCCCC(F)(F)F)N1CC(N(C(COC(CC)(C)C)=O)C)C2(C1)CC2 77730,C1(C(N(CC(C)(CO)CO)C)=O)CCN(C(=O)C2CCCS2)O1 77731,C#Cc1cncc(CNc2ncc(OCc3ccccc3)cn2)c1 77732,C(c1cscn1)=CC(=O)NCC1CCC1NC(c1coc(C2CCC2)n1)=O 77733,C(=O)(C1=CCN(C(=O)CN2C(=O)CNC2=O)CC1)NC(C)CC1CCC1 77734,N1(C(CN2CC(C)C2)=O)CC2CCC(NC(=O)CCC3(C)CC3)CC2C1 77735,C1(C)(C(=O)NC(CC)C(=O)NCC(F)Br)CC2(CCC2)C1 77736,c1(C(=O)NCCC2CCN(C(=O)CCC=CBr)C2)cnc2c(c1)CCOC2 77737,CC(C(=O)NC1(CNC(c2cn(CC(N)=O)nn2)=O)CCOCC1)S(N)(=O)=O 77738,C1(C)(C(N(CC(C)(C)NC(C2C(C(=O)OC)CC2)=O)C)=O)CCOC1 77739,CC1CN(C(=O)CCOCCN(C(=O)C(c2ccn(C)n2)C)C)CC1C 77740,c1(C(c2nnnn2C2CCCC2)NC2(C)CCCC2)cc2ccccc2nc1O 77741,c1(C(=O)NCCn2cc(C(CC)N(C)C)nn2)cc(C)c2nc(C)nn2c1 77742,c1(C(=O)NC2(CCNC(C(COC)OC)=O)CCC2)cn2cnnc2cn1 77743,Cc1cc(=NC(=O)C(=O)NC2CC3CN(C(=O)CCc4ncc[nH]4)CC3C2)[nH]o1 77744,Cc1cc(=NCc2nc3ncccc3o2)[nH]c(N(C)Cc2ccc(Br)cc2C)n1 77745,C(C)(CC(=O)O)(c1n(CC=C)nnn1)NCCC1(c2ccccc2)CCCO1 77746,C1(C)(NC(C(n2c(C)ccn2)C)=O)CCCN(C(=O)C2=COCCO2)C1 77747,Cc1ccc2c(c1)C(C(=O)N1CCN(C(c3cc(=O)cc[nH]3)=O)CC1CCO)C2 77748,c1(OC)ncc(Br)c(=NC(CNC(C2COCCO2)=O)C(C)C)[nH]1 77749,N1(C(CC2CC(C)C2)=O)CCC(C(C)C)CC1CNC(=O)Cn1cccnc1=O 77750,N1(C(c2cn(C)nn2)=O)CCN(C(=O)C=CC2CC2)C(c2ccnn2C)C1 77751,N(C1CC2(CCCC2)c2ccccc21)C(C(CC)NC)=O 77752,c1(C(=O)NCC(CNC(CCCC(=O)OCC)=O)OC)cnn2c1CCCC2 77753,c1(CC)nc(NCC(C2CC2)NC(=O)C(C)(O)C(C)C)c2ccsc2n1 77754,C1(CNC(C2ON=C(C)C2)=O)(CNC(c2[nH]ccc2C2CC2)=O)CCCCC1 77755,C1(C(N(C2(C)CCCC2)C)=O)CN(C(C2CC(C3CC3)C2)=O)CCO1 77756,C1(NC(c2cc(F)c(OC)c(Cl)c2)=O)C(C#N)CCC12CCOCC2 77757,N1(C(N(C2CC2C=CCOc2ccc(Cl)c(Cl)c2)C)=O)CC(C)(CO)CC1(C)C 77758,N1(C(CCCC)=O)CC2(CCCC2)C1C(N1CCC2C(C(N)=O)C2C1)=O 77759,C(C(C)(C)CCNC(c1csc(CO)n1)=O)NC(Cc1c(C)ncs1)=O 77760,c1(OCC)cccc(CC(=O)NCCCCN(C)C(c2c[nH]ccc2=O)=O)n1 77761,C1(CNC(CCOCCCOC)=O)CC2CCC1N(C(=O)CC1CC3CC3C1)C2 77762,N12CCCC(C3CN(C3)C(=O)C3(CC3)C1=O)C2.C1(COC(C)C)C2CCCCC12 77763,c1(CC(=O)NCC(CC)N(C(c2c(CC)c[nH]n2)=O)C)cncc(C)c1 77764,CCCC(C)C(=O)NCC1(C(C)NC(c2cc(N(C)C)ccn2)=O)CC1 77765,C12(CC(=O)N(C)CC3(C)CC3)CCC1CN(C(C1(C3(O)CCC3)CC1)=O)C2 77766,CC(C)C(C(=O)NN1CC(C)C1)n1ccc(C2CC2)n1.C1(C(C)(C)C)N=N1 77767,C(C(CNC(c1n[nH]c2c1CCC2)=O)S(C)(=O)=O)NC(C1OCC(C)(C)C1)=O 77768,N1(C(c2cn(C)nn2)=O)CCC2(NC(=O)CC(F)(F)C(F)F)CCCCC12 77769,N1(C(C2(NC(C)C)CC2)=O)CCC(C2CCN(C(c3coc(O)n3)=O)CC2)C1 77770,C12(C(=O)NC(C3CCN(C(=O)CC4CCOC4=O)CC3)C)CCOC(C)(C1)C2 77771,c1(N2CCC(OC(C)C)C2)nc(N2CCC(C3(C)CC3)C2)c2[nH]ccc2n1 77772,C(=O)(C(C)CCC(C)(C)C)N1C(C(=O)NC(CC#C)CC#C)CCOCC1 77773,c1(-c2nc(C(CC)O)nn2-c2ccc(Cl)cc2)ccc2ncccc2c1 77774,C1(C2CN(C(C3CCCO3)=O)C2)(NC(C2CCN2Cc2ccccc2)=O)CC1 77775,c1(CC(=O)N(C2CC(CCNC(CN(C)CS(CC)(=O)=O)=O)C2)C)nnc(C)s1 77776,c1(C(N2C(CNC(CCCOC(C)C)=O)CC(O)C2)=O)nccn2ccnc12 77777,n1(CC)ncc2c(C(=O)NCC(O)CNC(=O)C(C)(C)CO)cc(C3CC3)nc12 77778,c1(C(=O)NCC2N(C(C(C)OC)=O)CCN(C)C2)cccc2ccccc12 77779,Cc1ccc(CCNC(C2(C)CCN(C(c3ccc(Cl)cc3)=O)C2)=O)cc1 77780,N1(CC)CC(CN(c2nc(C)ncc2F)C(C2CCNCC2)=O)OC(C)C1 77781,CC(C)(F)C(C)(F)C(=O)NCC1(O)CC(CNC(c2cc(O)nc(Cl)c2)=O)C1 77782,c1(CCC)n[nH]cc1C(=O)NC(COC)C(=O)NC(C)CO 77783,n1(C(C)C)c(C2CCCN(C(C3C4CC3N(C)C4)=O)C2)nc2ccccc12 77784,c1(C(N2C(C(C)(C)NC(C3C(OC)CCCC3)=O)CCC2)=O)ccc(C)c(F)c1 77785,c1(CNC(CCC2(NC(C3CCC(CC)O3)=O)CCC2)=O)cc(C)nc(O)c1 77786,N1(C(C(C)(C)C2CCN(C(=O)NC3CC3)C2)=O)CCC(C)(CCO)C1 77787,c1(C(=O)NC2CN(C(CC(C)F)=O)CC2(C)C)c2ccccc2nn1C 77788,c1(C(=O)NCC2(S(N)(=O)=O)CC2)c[nH]c2ccc(C3=CCOC3)cc12 77789,N1(C(C(C(C)SC)O)=O)CCC(C)(CNC(C2CC(OC(F)F)C2)=O)CC1 77790,c1(C(C(=O)NCCOCC)N(C)CCC2CCCCC2)c(Br)cnn1C 77791,Cc1cc(C)n(C(C)CC(=O)NC2C=CCN(C(=O)CSc3cn[nH]c3)C2)n1 77792,Cn1nc([N+](=O)[O-])cc1C(=O)NCC1CN(C(C2CCS(=O)(=O)CC2)=O)C2CC12 77793,C1(N(C(=O)Cn2cc(C3CCCC3)nn2)C)CNC(=O)C12CC2 77794,S(=O)(=O)(c1ccc(F)c(C(F)(F)F)c1)NCC1CCC(NC(C(N)=O)=O)C1 77795,c1(C(C)C)cccc(C(=O)NC2CC2NC(=O)C(c2ccc(Cl)s2)C)c1 77796,C(=O)(CC(CC(C)C)NC(=O)C(F)(F)CCCC)NCC(CC#C)(C)C 77797,Cc1cc(C)n(CCNC(=O)C(CC2CC2)NC(=O)COc2cnn(C)c2)n1 77798,c1(C(N2CCCN(C(C(C=C=C)C)=O)CC2)=O)cc(OC)c(OC)cc1F 77799,Cc1cnc(C(=O)NCC(O)CN(C)C(c2nocc2C(C)(C)C)=O)c(F)c1 77800,N1(C(C(=O)NC(C)C)=O)CC2CCN(C(c3ccn4nccc4c3)=O)CC2C1 77801,N1(C(c2c(SCC)cccn2)=O)CCCC(C2CCN(C(=O)CCOC)CC2)C1 77802,c1(NC(=O)NC2CN(C(=O)OC(C)(C)C)C2)conc1C1CC1 77803,C1(CNC(c2c(SC)snn2)=O)CC2(CO1)CN(C(C1CC=CC1)=O)C2 77804,N1(c2cnc(C(C)=O)c(C)n2)CCCC1C1CCCCN1C(=O)C(C)CO 77805,C1(CC(=O)N(C(C)CCNC(=O)COCCN(C)C)C)CCC12CCC2 77806,Cc1ncnc(C)c1OCC(=O)NC1CCC(NC(C2CS(=O)(=O)CCO2)=O)C1 77807,N1(C(C2CCC(=C)CC2)=O)CCCC(C)(C)C1C(N1CC(CN=[N+]=[N-])C1)=O 77808,O=C1NC(C2CCOC2)C(=O)N1CC1CC2CCC1CC2 77809,c1(OC)oc(C)nc1C(=O)NC(C)CC(C)NC(c1c[nH]nc1C(C)(C)C)=O 77810,CCC(C)(C#N)C(=O)N(C)CC=CC(N1CCC(C)CC1C)=O 77811,C1(C2CN(C(=O)CCc3ccc(C#N)s3)C2)(NC(C2(c3cn(C)nc3)CC2)=O)CC1 77812,Cn1cc(Cl)c(C(=O)NCc2ccc(CC(C)NC(C34CC(F)C3C4)=O)cc2)n1 77813,C1(CC(=O)NCC2C(CNC(C(C)CC3CCC3)=O)C2(F)F)CC(O)C12CCC2 77814,C1(CNC(C(=O)NCc2nccc(-c3ccccc3)n2)=O)CNCCC1(F)F 77815,Cc1ccc(-c2cn(CC3C(CO)C3(F)F)nn2)nc1.N1(CC(=O)N)CCCNC1=O 77816,N1(C(COCC)=O)CCC(C(F)F)(CNC(c2cncnc2)=O)C1 77817,Cc1[nH]nc(Cl)c1C(=O)NC1CCC(NC(=O)CC(O)c2ccccc2)C1 77818,c1(C(=O)NCC2CN(C(c3ccc(OC)nc3F)=O)C2)c[nH]c2nc(F)ccc12 77819,C(=O)(CCCC(C)CC)N1C(C)CC(CC(N2CC(C(=O)OC)C2)=O)C1 77820,N(C(=NCCCCC)N1CCc2c(cc(F)c(F)c2F)C1)C(C#C)CCCOC 77821,CCCCC(CC)CC(=O)N1CC(NC(C2(CC3CC3)CC2)=O)C(C2CC2)C1 77822,N1(C(C(C)c2cc[nH]n2)=O)CCCC12CCN(C(=O)CC(C)(C)N(C)C)CC2 77823,n1(CC)nc(C)c(C(=O)Nc2c(N(C(COC(=N)O)C)C)ncnc2Cl)c1C 77824,c1(C(=O)OCC)cn(C)nc1C(N1CC(NC(=O)CN2CCC2C)C(F)C1)=O 77825,CCC(C)(C)CC(=O)N(C)CC1(O)CCN(C(c2ccc([N+](=O)[O-])s2)=O)C1 77826,c1(CC(=O)NCC(C2CC2)NC(=O)CCn2ccnc2)ccc(Cl)nc1F 77827,c1(C(=O)NCC(C)N(C(=O)C(C)CC(F)F)CC)ccnc2[nH]c(C)nc12 77828,Cc1cc(C(=O)NCC(CNC(=O)CC#N)CO)n(C(C)(C)C)n1 77829,n1(CC(=O)NC(Cn2cncn2)C(=O)NC(C)COCC)ccnc1C.CCC 77830,c1(C(=O)NC(C2CCN(C(C(C)OCC)=O)CC2)C(C)C)csc2nnsc12 77831,c1(CN(C(=O)C(C)OCCC(C)C)CC(C)NC(CSC)C)ccccc1 77832,n1(CCC)ccnc1C(F)(F)C(=O)N(CC(C)NC(=O)CC(C)C1CCCC1)C 77833,CCC(C)CC(CO)Nc1ncc(CN(C)C)cc1Br 77834,C1(NC(C(=O)NCCC2CC(OCC)C2)=O)CCN(C2CCCCC2O)CC1 77835,CCCCC(O)C(=O)NCCC1CCCN(C(c2ccc(C)c(OC)c2)=O)CC1 77836,N1(C(C2CCC(=C)CC2)=O)C(C(=O)NC(C)(CC)CO)CCC12CC2 77837,CCS(=O)(=O)CC(=O)N1CC2CC2C1C(=O)NCCCc1nnnn1C 77838,c1(C(=O)NCC2CN(C(c3cnn(CCC)c3C)=O)CC2C)cnc(C)c(N)c1 77839,c1(C(=O)OC)cccc(C(=O)NCC2C(C(=O)Nc3ccc(SC)cc3)C2)n1 77840,N1(C(=O)OC(C)(C)C)CCC2CC1CN(CNc1ccnn1C1CCCCC1)C2 77841,c1(-c2onc(CNC(=O)NC3CCCC=C3Br)n2)cccc(F)c1 77842,N1(C(C(c2cscn2)N(C)C)=O)CCN(C(c2cnn(C3CC3)c2)=O)CC(O)C1.C1CC1 77843,C1(CNC(c2nc(C(C)=O)sc2)=O)C2CN(C(=O)CC=C(C)C)CC12 77844,n1(C(C)C)ccc2c(N3CCC3(C)C(=O)NC(c3ccno3)C)ncnc12 77845,CC1CN(C(=O)CCC2(C)CC2)CC2(CCN(C(C3CCCN3C)=O)CC2)O1 77846,c1(C(N2C(C(C)NC(C(CC)c3ccccc3)=O)CCC2)=O)cc(C)nc(C)c1 77847,N1(C(Cn2c(C)nnn2)=O)CCCCC1CCC(C)(C)NC(C1CC1F)=O 77848,S(=O)(=O)(c1nc(C)cs1)NC(c1cccc(OC)c1)CO 77849,N1(C(CC=CC)=O)CCCC2CCN(C(C3CC4(CSC4)C3)=O)CC12 77850,N1(C(CCC2N(C(C3CCSCC3)=O)CCC2)=O)CC(CO)C2(CC2)C1 77851,NC(=NCCOC(F)F)NCCC1CC1.c1(C2C(C)C2)ccccc1 77852,C(CCS(=O)(=O)N1CC(O)CC1CN(C)C)C1N(C)CCC1 77853,c1(C(C)C)c(C(=O)N(CC(C)NC(=O)CC2COC(=O)N2)C)cnc2ncnn12 77854,C1(C(=O)OCC)COCCN1C(C1(C)CCN1C(c1cnccc1Cl)=O)=O 77855,Cc1cc(C(=O)NCC2CCCC(NC(C3CC3F)=O)C2)cc(S(C)(=O)=O)c1F 77856,CC1(C)CC(C(=O)NCC2(O)CCN(C(=O)CCC3NC(=O)NC3=O)CC2)=NO1 77857,CCCC(CCC)C(=O)N1CCOCC1CNC(=O)C(CCSC)NC(N)=O 77858,CCC(C)C(O)CC(=O)NC1(CNC(=O)Cc2ccc(F)c(Cl)c2)CC1 77859,C1(CC(=O)NC2CCCN(C(C)C)C2=O)(OC)CC2(CCOCC2)C1 77860,C(C)(CCN=c1[nH]cnc2cc(C3CC3)nn12)NC(c1c(C)nn[nH]1)=O 77861,c1(C(N(CC(C)O)CCNC(CC=C=C)=O)=O)[nH]nc(C(F)(F)F)c1C 77862,C(C(C)(C)C(=O)NCCc1cn(C)nn1)NC(C1CCC(C)C1)=O 77863,N1(C(CCC2CCN(C(CC3C(C)OCC3)=O)CC2)=O)CC2CCC2(C)C1 77864,C(c1cscn1)=CC(=O)NCCSCC(=O)N(CC#C)Cc1ccco1 77865,Cc1[nH]c(=N)sc1C(N1CCOC(CN(C(=O)CC2C=NN(C)C2=O)C)C1)=O 77866,N1(C(C2(C)N(C(C3C(OC)(OC)CC3)=O)CC=C2)=O)CCC(C)(C(C)C)CC1 77867,N1(C(C2CC(OC)C2)=O)CC2CC(O)C1C2NC(c1cccnc1N)=O 77868,Cc1ncc(NC(=O)CCc2nc(C3CC3)no2)o1.C12(CCC1)NC(=O)CO2 77869,N1(C(C(COCC)N=[N+]=[N-])=O)CC(C(=O)N(C(C)C)CC2CC2)CCC1(C)C 77870,c1(C(C)NC(=O)C(C)(C2CC2)N(C)C(c2cn(C)cn2)=O)cccc(O)c1 77871,c1(CC)nnc2n1CCCC2C(=O)N1CCN(C(c2cccn2C)=O)C(CO)C1 77872,C1(n2cc(-c3cccc(C)c3)nn2)CON(C(=O)C2CC(n3ccnc3)CO2)C1 77873,c1(CC)ncc(C(=O)NC2(C)CC(NC(C3CN(c4nncs4)C3)=O)C2)s1 77874,C(=O)(N1CCC(C(=O)OC)O1)C1N(C(C)C)CCC1.C12CC1C(=O)N2.CN=[N+]=[N-] 77875,C1(NC(C=CC(=O)OCC)=O)CC12CCN(C(C1(n3ccnc3)CCCC1)=O)C2 77876,c1(CC(=O)NC2CCN(C(c3n(CCOC)ncc3)=O)C2C)ccc(Cl)cc1F 77877,CC(CCC(F)(F)F)NC(C1C2CCC1(c1ccco1)C2)=O 77878,C1(NC(CCCSC)=O)(CO)CCN(C(=O)CC2CC(F)C2)CC1 77879,Cc1nc(O)sc1C(N1CCC(CN(C(=O)C=Cc2ccncc2)C)C1)=O 77880,N1(C(C2C(=C)C2)=O)CCC2(CCCN(C(=O)CC3(CO)CCCC3)C2)C1 77881,C1(CC(C(=O)NC(C)CC)N(C)CC2(OC)CCCC2)COC(C)(C)O1 77882,c1(OC)ccc(CCC(=O)NC2(OC(C)=O)CN(C(=O)C(C)C(C)O)C2)c(OC)c1 77883,C1(C(=O)Nc2cccc(CC)c2F)CC(C)(C)CCN1C(=O)C(C)c1cc[nH]n1 77884,c1(CC(=O)NCC2CC(NC(=O)Cc3cnc(C4CC4)[nH]3)C2)cncc(F)c1 77885,N1(C(Cc2cc(CC)no2)=O)CC(NC(=O)Cc2ccn(C)n2)CC12CCC2 77886,Cc1cc2c(cc1C)C(NC(C1(N3CCCNCC3)CCC1)=O)CCS2 77887,c1(CC(N2C(C(C)(C)OC)CCC2)=O)ccc2occc2c1 77888,c1(CNCCC(C)CC(C)(C)C)cc2nc(Cl)ccc2s1 77889,N1(C(C(C)CN(C)C(C23CCCC2C3(F)F)=O)=O)CCC2(CC1)CSC2.CCO 77890,C(=O)(C(O)CCCNC(=O)CCc1cccnc1)NC(CCC)c1nn[nH]n1 77891,C=C=CC(C)C(=O)N1CCCC1C(C)(C)C(=O)Nc1cnc(N(C)C)nc1 77892,C1(C(=O)NC2(CC)CN(C(C3CCN(C)C3)=O)C2)OCCN(C)C1=O 77893,C1(CNC(c2csc(C)c2C)=O)CN(C(C2CCOC2)=O)CC(C)(C)C1 77894,C1(NC(C2(C=C)CCC2)=O)CC(O)CN(C(c2ccc(OC)c(C)c2)=O)C1 77895,c1(C(=O)NCCCN(C(CNS(CCOCC)(=O)=O)=O)C)ccc(C)cc1CC 77896,C1(NC(C2CC=CCN2C(=O)Cn2cccnc2=O)=O)CC12CCCCC2 77897,c1(C(=O)NC(CCCNC(COC(CC)C)=O)C)nccc(Br)c1O 77898,c1(OC)cc(C(N2CCCC(CN(C(=O)C=C(C)Cl)C)C2)=O)c(N)c(C)c1 77899,c1(NC(C(C2CN(C(c3n(C)nnc3)=O)C2)O)=O)cccnc1O 77900,N1(C(c2n[nH]c(C)c2C)=O)CCC(C)(CNC(C2CC2C(=O)NCCO)=O)CC1 77901,N1(C(CN2CCC(N(C)C)CC2)=O)CC=C(CNC(c2cnn(C)n2)=O)CC1 77902,C1(CNC(CCC)=O)CN(C(=O)C(O)C2=CCCCC2)C2CCCC2O1 77903,C(=O)(C(F)CC(C)(C)NC(=O)C(C)c1ccco1)Nc1cccc(C#C)c1 77904,C1(CCC=C)(C(=O)NCc2cnn(C)c2)CN(C(C2CCO2)=O)C1 77905,Cc1[nH]c2ccccc2c1C(=O)NCC(C)N(C)C(C1CCC(C)(C)C1)=O 77906,c1(CNC(C2CC2F)=O)cccc2c1CN(C(c1cc(O)ncc1F)=O)C2 77907,c1(C(N2C(CC(=O)OC)COC(C)(C)C2)=O)ccc(Cl)cc1N=[N+]=[N-] 77908,C1(C#N)(C(=O)NCCc2c(C(N(CC(C)(C)CO)C3CC3)=O)c[nH]n2)CCCO1 77909,C=CCCCCC(=O)NC(C)CCCCNC(C1CCCN1c1cnccn1)=O 77910,NC1CC2(CC(CNC(C3(O)CCNCC3)=O)C2)C1 77911,C1(C)(CNC(Cn2nnc(C(C)(C)C)n2)=O)CN(C(=O)CC2CC(F)C2)CC1C 77912,C(=O)(C(CO)C(C)(C)C)NCC1N(C(CCOCc2ccc(OC)cc2)=O)CC1 77913,Cc1cc(C(N2CC(CNC(C3COC3)=O)CC2C)=O)c2nc(C)n(C)c2n1 77914,CCC(C)(O)C(=O)NCC1CCN1C(=O)CCc1ccc(C(F)(F)F)nc1 77915,c1(COC)ccsc1C(N1CCC(NC(c2ccc(C(C)(C)C)[nH]2)=O)C1)=O 77916,c1(OC)c(NC(=O)C(F)C2CC(NC(C3CC4(CC4)CO3)=O)C2)cccc1F 77917,c1(NC(C2C(C)(C(=O)OCC)C2)=O)ccc(Br)cc1Br 77918,C(=O)(CC(C)CC(=O)NCC1(NC(c2ccc(Br)cc2C)=O)CCC1)OC 77919,c1(C(=O)NCC23OCC(NC(CC(C(C)C)O)=O)(C2)C3)cc(Cl)c(F)cc1F 77920,CC1CC(C)(C)CN1C(=O)COC1(C)CN(C(=O)C=Cc2cc[nH]n2)C1 77921,c1(CC(=O)NCCC2CCC(NC(CC(C=C)C)=O)C2)cn2cccc(C)c2n1 77922,Cc1cc(N2Cc3nn(C)c(N)c3C2)nc(=NCCn2ncc(Br)n2)[nH]1 77923,C(=O)(CCC(F)(F)C(F)(F)F)NCC1CN(C(c2c(C)cc(O)nn2)=O)C1 77924,N1(C(c2cc(SC)oc2)=O)CC(C2CCN(C(C3CCOC(C)(C)C3)=O)CC2)C1 77925,C(CC(=O)CCN(CC)CC)NC.C(C(=O)NC(C)COC)NC 77926,C1(C(NOC(C)(C)CO)=O)CC1C1CN(C(C2CCCCCC2)=O)C1 77927,CC(CC(=O)NCCCC1CCCN1C(=O)CCN1CCCC1)P(C)(C)=O 77928,C(CC(C)CCCC(C)C)NC(c1n(CCCC)nnn1)c1ccnn1CC 77929,c1(C(=O)NC2CCC(C(N3C(C#C)CC3)=O)C2)ccc(F)cc1F 77930,N1(C(c2ncc(OCC)nc2)=O)CCC2(NC(=O)CCc3c[nH]c(=N)[nH]3)CC2C1 77931,C(C(N=[N+]=[N-])C(=O)NCc1ocnc1C(=O)NOC)OCC 77932,C#CCC(CC(=O)N(C)CC1(N(C)C)CCC1)NC(=O)CC(C)C(F)F 77933,C#CC1(CNC(=O)CC2CCC(NC(C3CC4(CCO3)CC4)=O)C2)CCOCC1 77934,c1(C(=O)NCCC(CNC(C2N(C)CCC2)=O)O)cc(N)c(O)c(F)c1 77935,C1(NC(c2cc(O)ncc2F)=O)CC2CCC1CN2C(C1CCCC1)=O 77936,N1(C(COCC#C)=O)CCC(CO)(NC(c2coc(C(N)=O)c2)=O)C1 77937,C1(CCC)CCCN(C(=O)C#CCNC(C2CC(=O)N(C)C2)=O)CC1 77938,CS(=O)(=O)C1CC(C(=O)NCC2(C)CCN(C(c3[nH]ccc3C3CC3)=O)C2)C1 77939,C(=O)(C(C)(C)C)NCCC(=O)NCC1C(NC(C(C)=C(CC)C)=O)C1 77940,C1(C)(COC)CCCC1NC(=O)CN1CCC(NC(=O)CC(C)=C(C)C)C1 77941,C1(C(C(=O)NCCC=C=C)C)CCN(C(=O)Cc2noc(C)n2)CC1 77942,c1(CC)nnc(CN(C)C(C2COCC2NC(=O)C(COC)OC)=O)o1 77943,C1(C(N2CCN(C(CSCCCC)=O)CC2CF)=O)COC2CCCCC12 77944,c1(C(N(CCOCC#C)C)=O)coc(C(C)NC(C2CCC(=O)C2)=O)n1 77945,c1(N(CCC(=O)NC)C(C2(C)CCC2)=O)ncnc2sccc12 77946,c1(C(N2CCC(OCCNC(C3CC(SC)C3)=O)C2)=O)cc2cc(Cl)cnc2o1 77947,CN1CCC2(CCN(C(C3CC(CC(=O)O)C3(C)C)=O)C2)C1=O 77948,C1(NC(C(C)n2ccnn2)=O)CC(CNC(C2(C3CC3)CC2)=O)C1(C)C 77949,N1(C(=O)Nc2cnc(-c3ccccc3)s2)CCC(F)(C(c2ccccc2)C2CC2)C1 77950,c1(C(N2CCC(N(C(=O)C(c3ccc(C)s3)C)CC#C)C2)=O)nc(CC)oc1C 77951,Cc1cc(N)n(CC(=O)NC2CN(C(=O)CN(C3CCSC3)C)CC2C)n1 77952,C(=O)(CC(CC)C(C)(C)C)NC(c1cccnc1)C(N1CC(SCC)C1)=O 77953,C(=O)(C(C)(C)C(=O)NCCCCCCNC(C1CCN(C)S1(=O)=O)=O)OC 77954,N1(C(c2c(OC)nccc2)=O)CC(NC(=O)CCc2ccn(C)n2)CC12CCC2 77955,C(C)(CN=c1[nH]c(N2C3CCC2CC(CC(F)(F)F)C3)nc(=N)[nH]1)OCC=C 77956,c1(CC)nc(C)cc(=NC(CNC(=O)C(F)C(C)C)C2CC2c2ccccc2)[nH]1 77957,C1(C(C)NC(C(n2ccc(C)n2)(C)C)=O)CCCCN1C(=O)Cc1cnccn1 77958,Cc1cc(F)cnc1-c1cn(Cc2ncoc2CNC(c2cc(Br)n[nH]2)=O)nn1 77959,C1(CCCC)(C(N2CCC(C(C)OCC)C2)=O)CCC(=O)CC1 77960,c1(C(N(C)C)=O)cccc(CN2CCCCC2CNC(=O)CC2CC(=O)N2)c1 77961,c1(C(C(=O)N(CCN(C)Cc2cn(CCCCCC)nn2)C)C)cccc(F)c1 77962,C1(F)(C(=O)NC(CCC)(C)C)CCN(C(c2cc(C)co2)=O)C1 77963,N1(C(CC(CN(C)C)O)=O)CC(C)(C)CC1CNC(c1cc(O)nc(O)c1)=O 77964,c1(NC2C(CC)C2)ncccc1S(=O)(=O)NCc1nc2ncccn2n1 77965,C(CCCC(C)(C)NC(=O)C(C)NC(C)C)NC(CC1CC(OC)C1)=O 77966,c1(C(C)=O)ccc(NC(C2CC(F)CN(Cc3ccc(Br)s3)C2)=O)c([N+](=O)[O-])c1 77967,c1(C(N(C(CNC(C(CC=C)C)=O)C)C)=O)c[nH]c2cccc(Cl)c12 77968,CC1(C)CNCCC1N1CCN(Cc2cc(Cl)ncc2Cl)CC1 77969,c1(C(N2CC(C(C)NC(c3cc(CF)on3)=O)OCC2)=O)cc(Cl)c(O)c(Cl)c1 77970,C1(O)(CNC(CC(C)F)=O)CCCN(C(c2ccc(C(F)F)cc2F)=O)CC1 77971,CCC(CC)C(C)N=c1nc(N2CCC(CCCO)C2)c2[nH]ccc2[nH]1 77972,CC1CN(C(=O)C(C)N(C)C(C2CC(=O)OC2(C)C)=O)C(C)C1C 77973,N1(C(=O)OC(C)(C)C)CC2CC2(C(=O)NC2CCN(Cc3cccnc3)CC2)C1 77974,c1(C(N2C3C(NC(=O)C=CC4CCC4)CC(C3)C2)=O)ccc2ccncc2n1 77975,c1(N2CCN(C(=O)Nc3cc(C)ncc3Cl)CC2)cccc2nsnc12 77976,C=Cc1cncc(C(=O)NC2(CO)CCCN(C(=O)CN(C)C)C2)c1 77977,N1(C(C2C(CC)CCC2)=O)CC2C(CNC(C3CCC(=O)N3C)=O)C2C1 77978,N1(C(C2CCN(CC)C2)=O)CCOC(CCCNC(=O)CSC2CC2)C1 77979,N1(C(CCc2c(C)noc2Cl)=O)CCC2(CCN(C(=O)CCn3ccnc3)C2)C1 77980,N1(C(c2c(C)ncnc2)=O)CC2CCC(C1)C2NC(C1(C)CC2CCC(C1)S2)=O 77981,c1(NC(c2n(CCC)nnn2)C(C2CCCC2)OC)ccc2c(c1)OC(F)(F)O2 77982,c1(CC#N)cccc(C(=O)NC2CC(C(=O)NCC3NC(=O)NC3=O)C2)c1 77983,N1(C(c2cc(C)on2)=O)CCCC(O)(CN(C)C(c2ccc(C(C)C)nc2)=O)C1 77984,C(=O)(C(C(=O)c1ccccc1)NC(=O)OC(C)(C)C)OC1(CCCC)CC1 77985,C(=O)(C1=CC2C=CC1C2)NC(C1CCCN1C(c1cc2ccccn2n1)=O)C 77986,c1(OCC(=O)N(CCNC(c2ccc(C(C)(C)C)o2)=O)CC)ccc(Cl)nc1 77987,C(=O)(CC(O)CC(C)C)NC(C(=O)NC(CC(=O)OC)C)COC(C)C 77988,c1(C(N(CC(C)C)CCC)=O)cccc(CNC(=O)CSCC(=O)OC)n1 77989,CCC(C)C(O)C(C)C(=O)NCC(C)(C)CC(=O)NCC(N)=O 77990,CCC(CC(F)(F)F)NC(=O)CC(C)N(C(=O)Cc1cncnc1)C 77991,c1(CNC(=O)NCC(C2CCCC2)C)cccc(F)c1O 77992,C(=O)(C(C)CC(C)CC)N1CCC(OCC(=O)N(C(C=C)C2CC2)C)C1 77993,CC1CC2(CCN(C(=O)C(N3CCCC(c4ncco4)C3)=O)C2)CO1 77994,Cc1cc(O)c(Cl)cc1C(=O)NCCCCNC(=O)C(C)CC1CCC1 77995,N1(C(C2CC3(CCC3)CN2C(=O)CC2CSCCO2)=O)CCc2nnnn2CC1 77996,C1(CNC(C23OC(C)C(CC2)C3)=O)CC2(CO1)CN(C(C1CC(O)C1)=O)C2 77997,C#CC1CCN1C(C1CC(CCNC(=O)CC2(NC(C)=O)CC2)C1)=O 77998,c1(SC)sccc1C(N1CCCC1CNC(c1ncoc1C(F)(F)F)=O)=O 77999,c1(C(=O)NCCn2c(C)nnn2)ccc2c(c1)CCN2Cc1ccco1 78000,C1(C(C)C)CC(CNC(C2(CN)CCCO2)=O)CCO1 78001,c1(CC(N2CCCC(NC(C(CC)O)=O)C2)=O)ccc(Cl)c(Cl)c1 78002,C=C(C)C1CN(C(=O)CCNC(C2CC2(C)C(C)C)=O)CCO1 78003,N1(C(c2ccnc(C)n2)=O)CCC2(CC(NC(=O)Cc3cccc(C)c3Cl)C2)C1 78004,CCCCCC(CC)C(=O)NCC1CN(C(C23CC(C2)C3)=O)CCCO1 78005,c1(C(C(=O)NC(CC)C)N(CCC(N)=O)C)ccn(-c2cnn(C)c2)c1 78006,Cc1n[nH]cc1C(=O)NC1(C(=O)NCC2(F)CCOC2)CSC1 78007,N1(C(C)=O)CCOC(C)C1C.C(=O)(C(C)n1ccnc1)N(CC(=O)ON)CC#C 78008,N1(C(CC=CC=C)=O)CCC(C=C)(C(=O)NCCC(C)CCC)CC1 78009,c1(COC)cc(C)c(C2CC2)cc1Cl.C12(C(=O)OC)CCN(C1)C(=O)N2 78010,C1(NC(CC(C)OC)=O)CN(C(=O)CCCc2cnccn2)CC12CCC2 78011,C1(CNC(C(=O)NC(c2ccccc2F)CC)=O)CCC2(CC1)CC(N)C2 78012,CC1(C)CCC(NC(C2(c3ncco3)CC2)=O)C(CNC(c2ccoc2)=O)C1 78013,C1(CC)(CC)CC(O)CN1C(C1CC(NC(c2c[nH]c(=N)o2)=O)C1)=O 78014,N1(C(C2CC23CCC3)=O)CCC(N=c2cc(C3CC3)nc(C3CC3)[nH]2)C1 78015,C1(CC)CN(C(=O)C(CCOC)OC)CCN1C(c1ccc(O)c(Br)c1)=O 78016,C1(NC(C(CO)NC(C(CCC)NC(N)=O)=O)=O)CCCC(O)CC1 78017,C1(C(C)C)CCC(C(=O)NC2COCC2NC(=O)CC2COCCO2)CC1 78018,C1(C(N2CCN(C(C3C(C)C3)=O)C(C)C2)=O)C(C)(C)CCCC1(C)C 78019,c1(C(=O)NC2C(CNC(c3cnc(O)s3)=O)CCC2)ccncc1Br 78020,c1(SC)cc(N2CC3(CCN3C(=O)CCc3cncc(C(F)(F)F)c3)C2)nc(C)n1 78021,S(=O)(=O)(c1cccc(Cl)c1)Nc1ccc(NC(c2ccc(C#N)cc2Cl)=O)nc1 78022,Cc1cc(Cl)ncc1CC(=O)NC(C1CCCCC1)CNC(=O)C1=COCC1 78023,N1(C(C2CCN(CC#C)CC2)=O)CC2CC(NC(C3CC(C)C3)=O)CC2C1 78024,C1(C(=O)NC(c2c(C)nccn2)C)Cc2ccccc2C1O 78025,N1(C(C=NOC)=O)CCN(c2ccccc2CNC(C2CCC2OC)=O)CC1 78026,c1(C(N2CCC(CO)C(O)C2)=O)cccc2[nH]nc(C3=COCC3)c12 78027,C(=O)(C(C)(C)Cc1cnn[nH]1)NCC1(CCNC(C(C=CC)O)=O)CC1 78028,C=CCC(CC=C)C(=O)NCC(CNC(=O)CCc1c(C)nc(O)nc1O)OC 78029,C#CC1C(C(=O)NCC2(NC(=O)COc3ccc(CC)cc3)CCCC2)C1(C)C 78030,c1(OCC(C)C)cc(Br)ccc1CNC(=O)NC(CO)C(=O)Nc1ccncc1 78031,C(=O)(C(CO)NC(=O)C(CC1CC1)NC(c1cc(C(C)=O)on1)=O)OC 78032,N1(C(C(C)CS(C)(=O)=O)=O)CCN(C(c2ccc3cnsc3c2)=O)CC12CCC2 78033,Cc1cc(-c2cscc2NC(c2ccnc(OC(F)F)c2)=O)cnc1O 78034,C1(CCNC(=O)Cc2ccsn2)CN(C(c2cocn2)=O)CCO1 78035,c1(C(N2CC3CN(C(COCCCCC)=O)C3CC2)=O)cnn2cc[nH]c(=O)c12 78036,c1(C(N2CC3(C(NC(c4cnc[nH]4)=O)CC3)C2)=O)noc2ncccc12 78037,Cc1cc(=NC(=O)C(=O)NCC=CCN2CCCC2)[nH]n1-c1ccc(Cl)cc1 78038,CS(=O)(=O)CCCCN(C1CCC12CCNCC2)C(=O)C(N)CN 78039,C1(CNC(c2snc(C)c2N)=O)C(C)CCCN1C(=O)CCC1CC1(Cl)Cl 78040,C1(C(=O)NCCC2CCCC2)CN(C(c2n[nH]c3c2COC3)=O)CC1C1CC1 78041,c1(C(=O)NCC2C(NC(CCn3ccc(C)n3)=O)C2)ccccc1N1CCC1 78042,N1(C(CN(C(=O)CCC2CCC(C)O2)CC)=O)CCC2=C(CCCC2)C1 78043,CC1(C)CCN(C(=O)C(F)C2CCC2)CC1NC(c1cc(C2CCC2)no1)=O 78044,C=C(C)CC(C)C(=O)NCC#CCNC(=O)CNC(=O)CC1CCCCC1 78045,C1(NC(c2c(SC)ccs2)=O)CCCCN(C(=O)CC(C)c2ccncc2)C1 78046,C1(C(=O)NC(CNC(C2COC(=O)N2C)=O)CO)(CC)CNC(=O)C1 78047,c1(NCC2(C)CC=CCC2)cc(=NC2CCCc3sccc32)[nH]c(C(F)(F)F)n1 78048,C1(CNC(C(C)OCC)=O)(Cn2cc(C3(O)CCOC3)nn2)CC12CCC2 78049,C1(OC)CC(C)CN(C(C2CC(F)C2)=O)C1 78050,c1(OC)c(NC(=O)CC2CCN(C(c3ccccc3I)=O)C2)cccc1F 78051,S(=O)(=O)(c1ccc(=NCc2cnn(C)c2Br)[nH]c1)NCc1ncc(C)cn1 78052,C(=O)(C1=NOC(C)(C)C1)N1C(CC(=O)N(c2c(CC)ccc(F)c2)CC)C2CCCC21 78053,C1(NC(c2ccc(F)c(CO)c2)=O)CCS(=O)(=O)C12CN(C(C1C=CCC1)=O)C2 78054,N1(C(C(c2ccc(OC)cc2)O)=O)CCC(O)C(C(N2CC3CCCC3C2)=O)C1 78055,CC1CCC(NC(=O)CCCC2CCCC2)CN1C(=O)Cc1cc(F)ccc1O 78056,c1(C(N2CCC3(CCN3C(=O)CC3CCCC(O)C3)C2)=O)ccc2[nH]ccc2c1 78057,N1(C(C2C(C)CCC2)=O)CCc2c(Br)cccc2C1.C12CCCC1C(=O)N2 78058,C(C1=CCCOC1)N(C(=O)CC1CCC(NC(c2cnc(C3CC3)o2)=O)CC1)C 78059,N1(C(C(C)=C(CC)C)=O)CCC2CCCC12CNC(=O)COc1cccc(C)c1 78060,C(CCNC(=O)Cn1nnnc1C(C)C)(C(C)C)NC(CN(S(CC)(=O)=O)C)=O 78061,C(C)(C)(CC(F)C(=O)N1CC(OCCOC)C1)NC(c1c(CC)ocn1)=O 78062,N1(C(C2(SC)CC2)=O)CC2CCC1CN2C(C1(CO)CC1)=O 78063,c1(C(N2CC(CNC(C3(CC#C)CCC3)=O)C2)=O)nccc(C)c1N 78064,c1(OC(C)C(=O)NCCCCN(C(=O)CC2COC(=O)C2)C)cc(Cl)cc(Cl)c1 78065,n1(CCC(=O)NCC(=O)NCC(=C)C)cc(-c2ccnn2C(C)C)nn1 78066,CC(C)(F)CCC(=O)NCC1CCCC1C(N1CCC(CCO)CC1)=O 78067,c1(C(=O)NCC2(O)CCN(C(C(C=C)(C)CC)=O)C2)cnc2c(c1)CCCC2 78068,c1(C(=O)NC2C(C)CN(C(=O)CC3SC(=N)NC3=O)C2)nc2ccccc2[nH]1 78069,N1(C(CN(CCC)C)=O)CCC2(CC1)CN(C(c1ccnnc1NC1CC1)=O)C2 78070,c1(C(=O)NCC(C)(C(C)C)NC(C2N(CC)CCC2)=O)ccc2ncnn2c1 78071,C1(C(=O)NC(c2cccnc2O)C)CC=CCC1NC(=O)CC1COCC1O 78072,c1(C(N(CC(C)N(C(C(C)OCCN(C)C)=O)C)C)=O)cccn1C 78073,C1(NCCNC(=O)NC(CCC)c2cccs2)CC12CCC(C(C)(C)CC)CC2 78074,n1(CCNC([N+](C)(C)C)=O)cc(C(=O)NC(COC)(C)C2CC2)cn1 78075,C#CCC(C)(C)C(=O)NCc1ncccc1C(=O)Nc1ccc(C(C)C)cc1 78076,O=C(C1=Cc2ccc(Cl)cc2OC1)NCC(CO)NC(c1ccc(O)cn1)=O 78077,n1(CC(N2CCC(CCCC)C2)=O)ccc2ccc(F)cc12 78078,c1(C(=O)NC2C(NC(C(CCCC)(C)F)=O)COCC2)cc2ccc(Cl)cc2o1 78079,C(=O)(CCC(C)CC)N1CC(CCNC(C2CC(=C)C2)=O)OCC1 78080,N1(C(c2ccc(OC)s2)=O)CCN(C(C2CCCC2C2CC2)=O)CC1C 78081,c1(C(=O)NC(C2CCCN(C(=O)C=CCF)C2)C)cnn2ccc(Cl)c(F)c12 78082,C(Cc1cccs1)(CC(=O)Nc1cnccc1C(C)C)NC(c1c(C)ccs1)=O 78083,CCC(CCCC(=O)N1CC2(CSC2)C1)NC(=O)C(c1ccnn1C)O 78084,N1(C(C2C(=C)CC2)=O)CCC2CN(C(c3c(Cl)ccc(OC)c3N)=O)CCC2C1 78085,CC(C)(CC(=O)NC1(C2CCN(C(=O)C(F)CC3CC3)C2)CC1)C(F)F 78086,C1(O)(CNC(c2ccc(O)nc2Cl)=O)CCCN(C(C2CS(=O)(=O)C2)=O)C1 78087,C1(CC)CCCC1(C)C(=O)NCCCNC(c1ccccc1OCC(N)=O)=O 78088,c1(N(CCN(C)CC2CCCCC2)C)nc(=N)[nH]c(=NCCN2CCCC(O)C2)[nH]1 78089,C1(C(=O)NCc2cc(Br)cs2)CC12CCN(C(c1ccc(Br)cc1F)=O)C2 78090,C(C(C(=O)N1CC(OC(C)=O)C1)NC(C1C=C(C)CS1)=O)OC 78091,N#Cc1ccc(NC(C2(CNC(=O)CCCCCO)CC2)=O)cc1C#N 78092,Cc1ncnc(C)c1OCC(N1CC2C(NC(c3cccc(F)c3O)=O)C2C1)=O 78093,C1(C(=O)NC23CN(C(CN(C4CCC4)C)=O)C(C2)C3)CC2(CCCCC2)C1 78094,c1(C(=O)NCC2OCC(CNC(CC3CC(=C)C3)=O)C2)ccc[n+]([O-])c1 78095,c1(C(=O)NCC(C2CC2)NC(=O)CN2CCCCCC2)cc2c(Cl)cncc2o1 78096,C(=O)(C1=CC2C=CC1C2)N1CC2C(CC(=O)NCC(O)C3(Cl)CC3)(CC2)C1 78097,N1(CCNC(Cc2c(C)nc[nH]2)=O)CCN(C(c2ccsc2)C)CC1 78098,Cc1cccc2c(C(=O)N(C3CC4CCC(C3)N4C(=O)C=CC(C)C)C)csc12 78099,c1(OC)cc(=O)n(C)cc1C(=O)NCCOC1CN(C(=O)C2=CCS(=O)(=O)C2)C1 78100,N1(C(c2cc(C)on2)=O)CCC(NC(c2cc(C(F)F)cs2)=O)C(O)C1 78101,C1(C(N2CCCCC(NC(c3c(C)c(N)n(C)n3)=O)C2)=O)CC2C=CCC(C1)C2 78102,N1(C(CCC)=O)CC=CC(C(N2CCC(OCCF)C2)=O)C1 78103,c1(C(=O)NCCC2(NC(CC3CC(=C)C3)=O)CC2)sc2ccccc2c1Cl 78104,n1(CCNC(=O)OC(C)(C)C)ccnc1SCC(C)(O)C1CC1 78105,c1(CN(C)C(c2ccccc2F)=O)ccccc1CNC(c1c[nH]nc1Cl)=O 78106,c1(C(=O)NCCC(C)N(C)C(C2CN(C)C2)=O)c[nH]nc1-c1ccccc1 78107,n1(CC=C)c(N2CCC(N3CCOC3=O)C2)nnc1-c1cccn1C 78108,c1(-n2ncc(C)c2)ccc(CNC(N2CCOC(C)(C3CC3)C2)=O)cc1F 78109,N#Cc1cnccc1-c1ccc(C(=O)NCC2Cc3ccccc3O2)nn1 78110,N1(C(C=CC(=O)OCC)=O)CCSCC1C(N1CCCOCC1)=O 78111,CC(C)CC(C)CNC(=O)CCN(C(=O)CC1CCCC(C)C1)CCO 78112,C1(N(C(C=C(C)C(F)F)=O)C)CN(C(=O)C(CCN(C)C)N(C)C)CCC1O 78113,CCC(=O)CCC(=O)NC(C)CCCC(=O)NC1CCN(CC)C1 78114,N1(C(=O)CC2CCCCCCC2)CC2CCN(C(C3CC4CC4C3)=O)CC12 78115,c1(C(N2C(CNC(C(C)Cc3ccccc3)=O)CCC2)=O)nc[nH]c2ncnc1-2 78116,O=C(CC1=CCOCC1)NC1CCC1NC(c1ccc(C2CC2)cn1)=O 78117,c1(C(=O)NCC2CCC(NC(CCSC)=O)C2)ccc(N(C)C)c([N+](=O)[O-])c1 78118,C1(CNC(C2(C(C)(C)OC)CC2)=O)CN(C(c2cc(C)c(C)o2)=O)CC1C 78119,Cc1noc(C(CO)NC(=O)CCNC(=O)CNC(c2ccco2)=O)n1 78120,C1(C)(C(=O)OC)CCCN1C(C1(C)CN(C(c2cc(Br)ccn2)=O)C1)=O 78121,c1(C(N2C(CNC(c3n(CC)ncn3)=O)CC(O)C2)=O)cc(Cl)c(Cl)cc1O 78122,C1(C)(CNC(CCOC(C)=O)=O)CCN(C(=O)C=Cc2cnn(C)c2C)CC1 78123,Cc1ccc(C(=O)NC2CC2NC(C2COCC2(C)C)=O)c(N)c1F 78124,c1(C(N2C(CCNC(C3C(C=C)C3)=O)CCC2)=O)ccc2c(c1)CCN2C(C)=O 78125,c1(C(N2CC(CNC(C3CCC4CC4CC3)=O)OCC2)=O)ccc(O)cc1O 78126,N1(C(CSCCOC)=O)CCC2(CC1)CC(NC(=O)CCC1CNC(=O)N1)CO2 78127,c1(CC)noc(CCCC(=O)NCC(C)N(C)C(c2nccn2C)=O)n1 78128,C(=O)(C1=Cc2ccccc2C1)N1CCC(CNC(C(CO)N(C)C)=O)C1 78129,C1(CC)CN(C(=O)C(N2CCCC2)C2CC2)CCC1NC(c1ccncc1)=O 78130,N1(C(CCC(=O)N(CC)CC)=O)CCC(NC(=O)C(C)(C)CO)C(C)(C)C1 78131,C1(C(=O)OC)CN(C(=O)C(=O)Nc2cnn(C(C)(C)C)c2)CC1(F)F 78132,C(=O)(C(C)CS(C)=O)NCCN(C(c1ccc(CC(=O)OC)cc1)=O)C1CC1 78133,O=C(C#CC1CC(F)(F)C1)N1CCCCCC(NC(=O)C=CC(F)(F)F)C1 78134,C(C)(C)(CCCNC(=O)C(C)(C1CC1)OC)NC(C1CCC(CC)O1)=O 78135,CC1CCCCC1(CNC(=O)CC1CC=CC1)NC(C1OCCN(C)C1=O)=O 78136,c1(C(=O)NC(CC)CNC(=O)C(C)(C)F)ncc(OC)cc1F 78137,N1(C(COCCCC)=O)C2CCC1C1CC1(NC(=O)Cc1ccsc1C)C2 78138,C#CCC(CC(=O)NC1(C2CCCC2)CC1)NC(=O)CCC(=O)OC(C)(C)C 78139,Cc1ccncc1C(=O)NC1(CCNC(c2occc2Cl)=O)CC1 78140,C1(CNC(c2cnccn2)=O)CCCCCN1C(=O)CC1COCCO1 78141,C1(NC(c2c(C)n[nH]c2)=O)CC(C(=O)Nc2cnc(C(C)C)nc2)C12CCOCC2 78142,C(=O)(C(CC)C(=O)N1CCC(N(C(=O)CSCc2cccc(C)c2)C)C1)OCC 78143,C(=O)(CCC(C)SC)N(C(CNC(C1(C=C)CCC1)=O)Cc1ccccc1)C 78144,N1(C(c2cnc(Cl)s2)=O)CCC2CN(C(c3cccc4sccc34)=O)CC2C1 78145,c1(-c2nnc(C3(CC)CCCC3O)o2)cccc2c1CN(CCF)CC2 78146,N1(C(=O)C(Cl)=CCl)CC(NC(C2(c3cccnc3)CC2)=O)C(F)C1 78147,N1(C(c2cc(C)cc(Cl)c2)=O)CCCC(NC(=O)C(O)CCC(C)C)CCC1 78148,N1(C(CCC)=O)CCCC1C(=O)NC(C)CNC(=O)C=CCOc1ccccc1 78149,N1(C(c2cc3n(n2)CCO3)=O)CC23CCCCC2(C1)CN(C(C1CC(O)C1)=O)C3 78150,C12CN(CCO1)C(=O)NC2.C1(CN(C)C)CCCN(c2ccc(Cl)cc2)C1 78151,n1(CCC)nc(C)cc1C(=O)NC1CCCCC1NC(c1n[nH]c(C)c1C)=O 78152,C1(C(=O)NCCCNC(c2ccc(OC(F)F)cc2F)=O)C2CC3C(C2=O)C13 78153,Cn1ncc2c(NCC3CSC3)nc(N3CCOC(C4CCOC4)C3)nc12 78154,C1(NC(=O)NC(Cc2ccc(OC)c(OC)c2)C)C(C)OC(C)C(C)C1 78155,N1(C(CCCCC)=O)CCN(C(c2ccn(CCC(F)(F)F)n2)=O)C(C)C1C 78156,C#Cc1ccc(C)c(NC(c2ncn3c2CCC3)=O)c1 78157,c1(C(=O)NC2CC(C)(CNC(=O)CC3CCCC(O)C3)C2)cc2ccccn2n1 78158,CCN=C(NCc1noc(C2CCC2)n1)NCC1COC1 78159,C1(C(=O)NCCCCN(C(C)C)C)CCN(C(C2CC2(C)C(C)C)=O)CC1 78160,C(=O)(C1=CC(C)CC1)NCCC(C)NC(c1c(C)occ1C(F)(F)F)=O 78161,N1(C(C2C3CCC(=O)C3C2)=O)CCCC12CCN(C(=O)C(F)(F)CO)C2 78162,C1(CNC(C2C(C)C(=O)C2)=O)CCCN(C(=O)C(c2cscn2)N(C)C)C1 78163,C#Cc1ccc(Cl)c(C(=O)NC2CCCN(C(C3CCC(C(N)=O)C3)=O)C2C)c1 78164,C1(NC(=NCC2(P(C)(C)=O)CC2)NCc2cccs2)CCC2(C1)OCCO2 78165,CN1CC(C(=O)NCCC(F)Cn2cc(CO)nn2)CCC1=O 78166,N1(C(CCc2cnn(CCN(C)C)n2)=O)CCN(C(=O)CCN2CCC(F)C2)CC1 78167,C(=O)(C1=C(C)OCCS1)NC1C(OC)CN(C(=O)CN2CCC(C)(C)C2)C1 78168,C=CC(C)N=C(Nc1cccc(C(=O)OCC)c1)N1CCC(OCC2CC2)CC1 78169,C(=O)(CC1COCc2ccccc21)N1CC=CC(NC(C2(C)ON=C(C)C2)=O)C1 78170,C12(C(=O)NC3C(NC(CCc4n(C)ccn4)=O)CCOC3)C3C4C1C1C2C3C41C 78171,C1(O)(CNC(C(CC=C)c2ccccc2)=O)CCCN(C(=O)C(=O)NC(C)C)C1 78172,N1(C(c2cnn(C3CCOCC3)c2)=O)CC2(C1)CN(C(C1(Cl)CC1)=O)CCO2 78173,c1(C(N2CCC(O)(CCNC(CC(C=C)C)=O)C2)=O)cc(F)c(C(F)F)cc1F 78174,C1(NC(c2ccc3n[nH]cc3c2)=O)C2CC3CN(C(c4coc(Cl)n4)=O)C1C3C2 78175,CCC(CC(=O)NC(CNC(c1csc(-c2ccc(Cl)cc2)c1)=O)CO)C(C)C 78176,c1(C(=O)NCCOCCOCCOCCNC(C2CC2C2CC2)=O)nc(O)[nH]c(=O)n1 78177,c1(NC(CCc2n(CC)ccn2)C)ncccc1S(=O)(=O)NC1(CC)CCOC1 78178,C#Cc1cn(C)nc1C(=O)N(C1CN(C(=O)CC2CS(=O)(=O)C2)C1)C 78179,CC1CC(C(=O)Nc2cc(C3CCCNC3)no2)C(C)O1 78180,C12(CC(=O)NCCC(CC)C)CCC1CN(C(c1cc(CO)on1)=O)C2 78181,N1(C(C2Cc3ccccc3C2)=O)CC2(CCCCN2C(C2CCCS2)=O)C1 78182,c1(OC)cccc(-n2nnc(C(=O)NCC(CO)NC(=O)C(C)C(C)O)c2C)c1 78183,N1(C(C(C=CCCC)O)=O)CC2CCC(C1)N2C(=O)Cc1ccc(F)c(F)c1 78184,CCC(C)CCCCC(=O)N(CC(=O)NCCN1CC2CC2C1)CC 78185,c1(C(=O)NCC(CO)NC(C=Cc2ccc(OC)cc2)=O)cc2ncccn2n1 78186,C(=O)(C(C(C)C1CC1)N1CCN(C(C)C)CC1)NCCC(=O)OCC 78187,N1(C(c2c(C)oc(Cl)n2)=O)C2CCC1C(CNC(c1ccc(Cl)cc1)=O)C2 78188,N1(C(c2c(C)scn2)=O)CC(NC(c2ccnc(N3CCCC3)c2)=O)CCC1C 78189,c1(C(C)NC(=O)NCc2cccc([N+](=O)[O-])c2F)nnc2c(=O)[nH]ccn12 78190,C(=O)(CC(CC1CC1)NC(c1c[nH]cc1C1CC1)=O)N1C(C(N)=O)CC1 78191,C1(NC(COCCCCCC)=O)(CNC(c2ccsc2Cl)=O)CCCCCC1 78192,C=CCC(CC=C)C(=O)NC1CN(C(c2cncc(NC)c2)=O)CCC1C 78193,C(=O)(C(C)(C)C1CCCCO1)OC(F)F.CC1CN(C)C(=O)CN1 78194,C(C)(C)(CC(F)(F)F)NC(C(C)CN(C)C(c1cncc(C#N)c1)=O)=O 78195,c1(C(=O)OC)[nH]c(C)c(C(=O)N(C)CCN(C(=O)CCOCC2CC2)C)c1CO 78196,c1(C(=O)NCC2(F)CC(NC(c3ccc(N)cc3Cl)=O)C2)cnc2ccccn12 78197,c1(C(N2C(CNC(C(COC)C)=O)CCCCC2)=O)cccc2c1CCCCC2 78198,C1(NC(=O)C(c2ccc(I)cc2)F)COc2ccccc2C1=O 78199,c1(C(N2CCC(C)(C(=O)Nc3ccnc(CO)c3)C2)C)ccc(C2CC2)c(F)c1 78200,c1(C(=O)NCC(CN(C(C2(C#C)CCOCC2)=O)C)O)ccc(C)c2c1CCC2 78201,C(=O)(CC(CNC(=O)Cc1cccnc1F)OC)NCc1cc(C(=O)OC)no1 78202,C1(CCNC(=O)Cc2ccccc2)CCCCN1C(C1CC=CCO1)=O 78203,c1(C(=O)NC2CN(C(c3occc3Br)=O)CCC2(F)F)c(F)c(F)nc(F)c1F 78204,c1(-c2c(C(N=c3cc(C)o[nH]3)=O)c3c(cc2)OCO3)cc(S(C)(=O)=O)ccc1F 78205,C1(NC(C2CCCC(F)(F)C2)=O)CCC12CN(C(c1cnn(CCO)c1)=O)C2 78206,CCCCC(CC)C(=O)NCCC1(O)CCN(C(c2ccc(=NC)[nH]c2)=O)C1 78207,Cc1cc(CCC(N2CCC(CNC(=O)C(C)N3CC(C)C3)C2)=O)no1 78208,N1(C(c2cc(CC)[nH]n2)=O)CCC(C(C)(C)C)(CNC(C2C(F)(F)C23CC3)=O)C1 78209,c1(C(=O)NCC#CCNC(C(C)N2CCC2)=O)c[nH]nc1C(C)(F)F 78210,c1(-c2c(C(C)C(=O)Nc3cncc(C(C)(C)C)c3)cccc2)ccc(C#N)cc1 78211,c1(-c2cn(CCN(c3cccc(F)n3)C(C)=O)nn2)ccc(F)c(C)c1C 78212,C(=O)(CCCCCC(C)(C)C)N(C(C)CNC(=O)CCCn1cncn1)C 78213,c1(C(=O)NC(CN(C(c2ccon2)=O)CC)C)cn(C)c2c(cnn2C)c1=O 78214,c1(C(C(=O)OC)(C)C)cccc(NCCCN(C(c2ccncc2)=O)C(C)C)c1 78215,C1(NC(c2n[nH]c(C)c2Cl)=O)CN(C(C2(C3CCC3)CC2)=O)CCC1CO 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78406,C(C)(CSC)(C(=O)NC(C1CCC1)C)NC(C1C(OCC)CC1)=O 78407,N1(C(c2noc(C)c2[N+](=O)[O-])=O)CCCCC(C2CN(C(C3(F)CC3)=O)C2)C1 78408,C(CC(CC)C(=O)NCCNCC(=O)NCC(=O)NC(=O)NC)=CC 78409,N1(C(Cc2ccc(C(=O)OC)nc2)=O)CCCC(NC(=O)C(F)C(C)(C)O)C1C 78410,c1(C(=O)OCCn2ncc(C)c2)csc2ccc(F)cc12 78411,c1(OC)ccc2c(c1)C(NC(c1ccc(C(F)F)c(Cl)c1)=O)CCC2 78412,C1(C(=O)NCC2(OC)CN(C(C3CSCC(=O)N3)=O)C2)CCC2CCCCN12 78413,Cc1ccc(C(N2CCCCC2CC(=O)NC(CN(C)C)C(C)(C)C)=O)nc1C 78414,c1(CC(N2CC(C(C)NC(c3cc(C)n(C)n3)=O)C2)=O)ccc(F)c(Cl)c1 78415,C12(C(N)=O)CCCC1(C(=O)NC1CCCC1NC(=O)Cc1nnc(O)s1)C2 78416,C1(C(=O)NC2CCC2)COCCC12CN(C(c1ccnc(Cl)n1)=O)C2 78417,N1(C(c2cc(CC)ncn2)=O)CCCC(O)(CCNC(c2ccc(Cl)o2)=O)C1 78418,c1(-c2cnc(C#N)c(F)c2)ccn2cc(C(=O)NC3CCCC(F)(F)C3)nc2c1 78419,N1(C(C=C(C)c2cccs2)=O)CCC(CO)(NC(=O)CCN2CCOC2=O)CC1 78420,C(=O)(C1CCCc2sccc21)N1CC(C(C)NC(C2CCCO2)=O)OCC1 78421,C1(OC)CCC(C(N2CC(F)CC2CNC(=O)C(c2nc(C)cs2)C)=O)CC1 78422,c1(C(=O)NCCn2cccc2)cn(C2CCOC2)nn1 78423,C(CC(=O)N(C(C)CN(C(=O)C(C)n1cncn1)C)C)OCCC 78424,c1(OC)ccc(C(C)(C)C(=O)NC(C2CN(C(=O)C(O)CN(C)C)C2)C)cc1 78425,c1(C(N2CCCC(CC)C2)C(=O)NCC(=C)C)csc([N+](=O)[O-])c1 78426,c1(SC)cnn(C)c1C(=O)NC(C1CCN(C(=O)CCCCC2CC2)C1)C 78427,C(=O)(C(C)(C)CCCF)N1CCC(C2N(C(C3=CC(C)(C)C3)=O)CCC2)CC1 78428,C(=O)(C1CCCn2cnnc21)NCC(CO)NC(Cc1ccc(OC)cc1)=O 78429,c1(CC(=O)NC(CN(C(=O)C=CC2CC2)CC)C)cc(SC)nn1C 78430,c1(C(N2C(CNC(c3ccc(OC)c(C)n3)=O)CCC2)=O)c(C)cc(Br)cc1C 78431,CC1(C)C2CCC(C2)C1C(N1CC(NC(C2CC(O)C2)=O)C1)=O 78432,c1(NC)cc(C(F)(F)F)ccc1C(=O)NCC(O)CNC(=O)CSC(F)F 78433,c1(OC)ccn2cc(C(N3CC=CC3CNC(c3cc(Cl)c[nH]3)=O)=O)nc2c1 78434,c1(C(N2CCC(NC(c3nn(CC)c(O)c3)=O)C(C)C2)=O)c(N)cc(F)cc1Cl 78435,CC(C)C1=NOC(C(=O)NCCCC(C)(C)NC(C2(C)CCC(=O)NC2)=O)C1 78436,C1(NC(c2cnn(C)n2)=O)CCCCC12CCCN(C(=O)CN1CC3CC3C1)C2 78437,c1(CC(N2CC3C(NC(CC(CC)C)=O)C(CC3)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 78438,c1(C(=O)NC2CCC(CNC(C3C(C)(C)C3(F)F)=O)C2)cc(F)ccc1F 78439,c1(NCC)cncc(NC(=O)SC2CCCN2C(c2ccccc2COC)=O)c1 78440,C(=O)(C1=CNC2=NCCCC2=C1)N(CC(CO)(CO)NC(CSC(C)C)=O)C 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78459,c1(OC)cccc(CNC(=O)OC(C)(C)C)c1C.C12CCCN(C1)C(=O)C(=O)N2 78460,C(=O)(C#CC1CCCOC1)NC1(CNC(C(COC)CC(C)C)=O)CC1 78461,c1(OC)ccc(C(=O)NCC2CCC(C)CN2C(c2cnc(Cl)s2)=O)cc1O 78462,C(=O)(CC(C)CC(=O)N(C(CC(F)F)C(=O)NCC1=C(C)CCC1)C)OC 78463,N1(C(c2c(C)n3c(n2)scc3)=O)CCC2C1CCCN2C(=O)CC(C)P(C)(C)=O 78464,C12(C(=O)OC)CCNC1CN(C(c1cccc(C3(C)CCO3)c1)=O)C2 78465,CC1CC(=O)NCCN1C(c1c[nH]nc1-c1ccc(Cl)s1)=O 78466,N1(C(C23CC(CC(C)O2)C3)=O)CC2CCCC(C1)N2C(=O)CCn1cncn1 78467,c1(C(=O)NC(CCSC)C)cc(CNC(=O)CCc2nncs2)[nH]n1 78468,C1(N(C)C(c2cnnn2C)=O)CC2CCC(C1)N2C(C1CC1F)=O 78469,C1(C(=O)NCCC2CCCN(C(CCCCC#N)=O)C2)CC12CCC1(CC1)CC2 78470,S(=O)(=O)(CCC(=O)NC1CC(NC(c2ccc(Cl)c(N)c2)=O)CC1O)NC 78471,C1(C(N(CCNC(C(F)=CCC)=O)C)=O)CC(CC)=NO1 78472,CCC(C)CC(C(=O)NCCOC1CC1)NC(=O)Cc1ccc(O)cc1 78473,C1(NC(c2cc(OC)ncn2)=O)CCCN(C(=O)OC(C)(C)C)C1C 78474,c1(NC(CC2N(C(C3CCC(CC)O3)=O)CC2)=O)ccc2ccoc2c1 78475,C(=O)(CC(C)CC(C)(C)C)NCC(CC)(C)NC(=O)Cn1ccc(C(F)F)n1 78476,N1(C(C(CC)n2cccn2)=O)CCC(NC(=O)CCCn2ccnn2)CC1 78477,C12(NC(=O)C(C3CCOCC3)O)CCCC1N(C(=O)CCc1ccon1)CCC2 78478,N1(C(C23OCC(COC)(C2)C3)=O)CCC2CN(C(=O)C(O)P(C)(C)=O)CC2C1 78479,c1(C(=O)NCCNC(C(C(C)C)SCC)=O)ccc(C)c(C#N)c1 78480,c1(C(=O)OC)cc(NC(=O)NC(C2CCCC2O)C)c2c(c1)CCC2 78481,CC1CCC(NC(=O)C=C2CCCC2)CN1C(c1cc(Br)n(C)c1)=O 78482,c1(C(CNC(=O)NC(CC)C(F)F)C(C)C)ccc(F)c(F)c1 78483,N1(C(c2nc(CC)oc2)=O)CC2CN(C(C3CCOC3)=O)CC2C1 78484,N1(C(CC2(OCC)CCC2)=O)CC(OC)C(NC(=O)Cc2ccccc2)C1 78485,c1(SC)nc(NC2(CNC(=O)CC3CCC(O)C3)CCCC2)cc(C)n1 78486,c1(OC)cc(C(N2CCCC(SC)CC2)C(=O)NC2CCC2)ccc1S(C)(=O)=O 78487,C1(N(C(=O)CC2(CO)CCCCC2)CC)CCCN(C(=O)CC(O)CC)C1 78488,C1(CC=C)(NC(=O)CCN2CCCC2)CCN(C(C2(CSC)CCC2)=O)C1 78489,C1(CNC(=O)C=CCN2CCCC2)(NC(C2COC(=O)N2)=O)CCOC1 78490,c1(CC)cccc(C(=O)NC2(CC)CCN(C(C3CC3(C)COC)=O)CC2)c1O 78491,CC1CCN(C(=O)Nc2coc(Oc3ccccc3)n2)CC1Nc1ccccn1 78492,CC(C)CCCC(C)C(=O)N1CCC(C(C)NC(C2(C)COC(=O)N2)=O)C1 78493,CCC(C)(C(=O)NCC1CC(NC(c2cc(N3CCCCC3)ccn2)=O)C1)OC 78494,c1(N2C(CNC(C(C)C)=O)CC(F)C2)cc(-c2cccs2)ncn1 78495,c1(C(N2C(CNC(=O)C=CCN3CCCC3)CC(OC)C2)=O)cc2cnccc2o1 78496,c1(CN(C)C)cc(C(=O)NCC2CCCN(Cc3cnc(Br)s3)C2)ccn1 78497,C(=O)(C1=CCCC1C)N(CC(C)O)CCNC(c1ccc(C2CC2)o1)=O 78498,Cc1cc(C)c(CNC(=O)COc2ccc(C(C)(C)C)cc2)s1 78499,CC1CN(C(c2cnc(Cl)cn2)=O)CC(C)N(C(c2cc(F)ccc2O)=O)C1 78500,c1(CC)cc(C(N2CC(NC(C3C(C)C3C)=O)C(F)C2)=O)cc2c[nH]nc12 78501,n1(CC(N2CCC(c3c(C(=O)OC)nco3)CC2)=O)cc(C)c(=O)cc1C 78502,Cc1ccc(=N)[nH]c1C(N1CC(NC(=O)C(C)(C)c2cccs2)CC1C)=O 78503,N1(C(c2cnc(C)s2)=O)CCCN(C(c2coc(Cl)c2)=O)CC1CO 78504,Cc1nn(C(C)C)cc1C(=O)NCC1CC1NC(=O)C(c1ccc(F)cc1)F 78505,C1(NC(C(C)(C)OC(C)C)=O)CCCC(NC(c2cncc(C(C)(C)C)c2)=O)C1 78506,C(CC(=O)N1CC2CC1CN2C1CC1)(C(F)(F)F)c1ccc(-c2[nH]c(=N)sc2)s1 78507,CCC(O)C(C)C(=O)NCC1CN(C(=O)Cc2cn[nH]c2)CC1C(F)(F)F 78508,C1(CNC(C(c2ccnn2C)NC(C(C)NC(CC)(C)C)=O)=O)CCC(F)(F)C1 78509,N1(C(C(C(C)NC(CC(COC)(C)C)=O)C)=O)CCc2ccncc21 78510,N1(C(c2c(CC)noc2)=O)CC2(CCC2)CC1C(=O)NC(C)Cc1ccccn1 78511,C(CCC(C)CC(=O)NCCNC(c1cccc(O)c1F)=O)=C(C)C 78512,C(=O)(C1CCCc2nnn(C)c21)N1C(CN(C)C(c2n[nH]cc2Cl)=O)CCC1 78513,C1(F)(CNC(c2n(CC(C)C)ncc2)=O)CCN(C(c2nc(=O)n(C)[nH]2)=O)CC1 78514,N1(C(C(C(=O)O)C2COC2)=O)CCC(S(=O)(=O)N2CCCC2)C1 78515,c1(C(=O)OC(C2CC2Cc2c(OC(C)C)cccc2)=O)c(Cl)cccc1[N+](=O)[O-] 78516,C1(O)(C(=O)NC2CCC(CNC(c3c(C)ccnc3C)=O)C2)CCC(C)(C)CC1 78517,N(C(=NCC(C)(C)OC1CCOCC1)NCC1(C)CCCS1)C(C)C 78518,N1(C(C2CN(C(c3cncc(C=C)c3)=O)CC2C(C)C)=O)CCC(O)C(C)(C)C1 78519,CN1N=C(C(=O)NCC2(CC(=O)NCC3CCCCS3)CC2)CCC1=O 78520,N#Cc1ccccc1.N12CC3CC1C3NC(=O)c1cnccc1C2=O.C(F)F 78521,C(=O)(C1=CCCC1C)NCC1(COC)CCCN1C(=O)CCS(C)(=O)=O 78522,N1(C(C(=O)OC)=O)CCOCC1C1CC1.N12C(CC1C)C(=O)O2 78523,c1(CC2(C(=O)NCC3(C)CC(NC(C4(C)CCCS4)=O)C3)CC2)cccc(F)c1 78524,c1(C(=O)NCc2cc(I)c[nH]2)ccc(NC(c2ccncc2)=O)cc1 78525,c1(C(C)C)noc(CCCC(=O)N(CC(C)NC(c2ncc(Cl)s2)=O)C)n1 78526,C12(CNC(C3N(CCC)CCC3)=O)CC1CN(C(=O)COC1CC=CC1)C2 78527,c1(CC(C)C)ncc(CNC(C)Cc2cnc[nH]2)s1 78528,N1(C(C2(OC)CC2)=O)CCC(NC(C2(C(F)(F)F)CC3(CCC3)C2)=O)C(O)C1 78529,CC1(C)OC2CC(C(N3CC(NC(=O)CCCS(C)(=O)=O)C(O)C3)=O)CC2O1 78530,c1(CNC(c2c(C)snn2)=O)ccc2c(c1)CCC2NC(=O)C#CC(C)C 78531,N1(C(C=C(C)CN2CCOCC2)=O)CC2CCN(C(c3cn[nH]c3)=O)CC(C2)C1 78532,C(=O)(C(C1(C)CC1)NC(=O)C(F)OC(F)(F)F)NCC(C1CCC1)OCC 78533,N1(C(c2ccc(C#N)s2)C(=O)Nc2c(C)cc(F)cc2)C2CCC1CC(CO)C2 78534,N1(C(CNC(N)=O)=O)CC2CCN(C(c3csc(-c4cccs4)n3)=O)CC12 78535,CC(C(=O)NCCCn1nccn1)N(C(=O)C=CC(=O)NC1CC1)C1CC1 78536,Cc1ncncc1C(=O)NCC1CN(C(c2ccnc(Br)c2)=O)CCO1 78537,c1(OC)cc(C(N2C3CN(C(c4sncc4C)=O)CC23)=O)cc(OC)c1C 78538,N1(C(C=C(CC)CC)=O)CCC2(CCCC2NC(C2CCS2(=O)=O)=O)CC1 78539,C1(CC)(NC(=O)C(C)OCC(C)C)CCCN(C(c2cc(N)nc(Cl)c2)=O)C1 78540,c1(C(=O)NC(c2ccccc2)C(=O)NC(c2ccnn2C)C)ccc(C#N)cn1 78541,CN1CC(C(N2CCCCC2C2CCN(C(=O)Cn3[nH]cnc3=N)C2)=O)NC1=O 78542,C1(C(=O)NC(c2nocc2C(=O)N(CCF)C2CC2)C)CC=CCC1 78543,C12(C(=O)NC(CC(=O)O)CC3CCCCCC3)CCCN1S(=O)(=O)CC2 78544,c1(CN(C(c2c(COC)ocn2)C(=O)NCCCF)C)c(C)noc1CC 78545,Cc1nn(C)c2c1CNC(=O)CO2.c1(CC2(F)CCOCC2)ccc(Cl)cc1Cl 78546,C1(O)(C(N2C3C(NC(=O)CC4CCCC4O)CC(C3)C2)=O)Cc2ccccc2C1 78547,c1(C(=O)NC2C(NC(CCC=C)=O)CC2)cc(CN2CCCC2)ccc1F 78548,c1(OC)cc(C)cc(C(=O)NCC2(O)CN(C(=O)C3=COCCC3)C2)c1N 78549,c1(C(C(=O)NC(C)CC)N(CCCN(C)C)CCC)ncc(C)c(OC)c1C 78550,c1(C(N(C2CN(C(C(C=CCCC)O)=O)CC23CC3)C)=O)cc(Cl)c(F)cc1F 78551,C1(C)(NC(c2n(CC)ncc2)=O)CCCN(C(c2cc(C(C)=O)cnc2O)=O)C1 78552,C#CC1(C(=O)NCC2(CC)CCC2)CCN(C(=O)C(O)C(C)C)C1 78553,C(c1csc(C(F)(F)F)c1)=CC(=O)NCCC(=C)CNC(=O)CC1OCCC1C 78554,C1(CNC(c2c(C)snn2)=O)CC(NC(c2ccc(C3CC3)s2)=O)C(O)C1 78555,N1(CCC(=O)NC(CCC=C)CO)C(=O)COCC1=O 78556,C1(C(=O)NC2CCN(CCNC(c3c(C)n[nH]c3)=O)CC2)CC(C)CC(C)C1 78557,C1(COC)Cc2ccccc2O1.c12ccc(cc1)C(=O)NC1(c3cn-2nn3)CC1 78558,N1(C(c2cncc(CC)c2)=O)CC2(CC(NC(=O)CC(C3CC3)OCC)CO2)C1 78559,CC1(C)CCN(C(=O)COCc2nccs2)CC1C(=O)NC(c1ccco1)CO 78560,C(N=c1[nH]c(C)c([N+](=O)[O-])cc1Cl)C1CC(NC(c2c(CC=C)cccc2)=O)C1 78561,c1(C(=O)OCC)c[nH]c(=NC)nc1CN(C)Cc1ncc(Cl)n1C 78562,N1(C(c2ncn(C(C)C)n2)=O)CCCC(CN(C)C(c2ccc(F)cc2)=O)C1 78563,C1(C(=O)NCCCC2CCCN2C(C2SCCS2)=O)CCC2C(C1)C2(F)F 78564,C(=O)(CCS(=O)(=O)N(C)C)NC1(C)CC(NC(c2cc(CC)nn2C)=O)C1 78565,C1(CNC(Cn2ncc(C)c2)=O)CC2(CO1)CN(C(=O)C(N1CCCCC1)C)C2 78566,CC1CN(C(=O)CCc2cccnc2)CC(C)N(C(c2ccc(CO)cc2)=O)C1 78567,C(CC(C)C(=O)NCC1(NC(=O)CCCc2n[nH]c(=N)s2)CCCC1)OC 78568,N1(C(=O)C(c2ccccc2Cl)O)CC(NC(C2(O)CCC2)=O)CC12CCOCC2 78569,CC(=Cn1ccnn1)C(=O)NCCC1(NC(C2CCCN2N=O)=O)CC1 78570,Cc1cc(C(N2C(C(N3CC(CC(N)=O)C3)=O)CCC2C(C)C)=O)[nH]c1C 78571,C1(NC(C2N(C(CC)=O)CCCC2)=O)CC2(CCN(C(=O)C(C)(O)C3CC3)C2)C1 78572,C1(N(C(c2cccs2)=O)CC)CCCN(C(=O)CSc2ccccc2)C1 78573,C(=O)(C(C)(C)CCCOc1ccccc1)OCc1c(C)cccc1Cl 78574,c1(C(N(C)CC2CN(C(=O)C=Cc3ccco3)C2)=O)ccnnc1Cl 78575,N1(C(C2N(C(C(C)(C)N(C)C)=O)C3(CC2)CC3)=O)C2CCC1CN(C)CC2 78576,C(CCCCC(=O)NC1CCC1CNC(=O)CC12COC(C)(C1)C2)SC 78577,c1(CC(=O)NC2(CNC(C=CC(C)(C)SC)=O)CC(F)(F)C2)ccc(C)cc1F 78578,c1(C(C)=O)ccc(OCC(=O)NCC(CC(C)C)NC(C2C=C2C)=O)cc1 78579,c1(NC(C(c2ccccc2)C)=O)cccc(NCC(F)(F)F)c1 78580,c1(C(=O)NCC2(F)CC(NC(CCCCOC)=O)C2)cc2ccccn2c1 78581,C(=O)(C(O)CCCC)N1CCC(CC=C)(C(N2CC(Cc3ccoc3)C2)=O)C1 78582,c1(C(N2CCOCC(NC(C3(C)C=CCCC3)=O)C2)=O)ccc(C#N)cc1O 78583,N1(C(C2(C(=O)NC)CCC2)=O)CCCC(C2CC2NC(C2CC23CCC3)=O)C1 78584,N1(C(CSSC)=O)CC(CNC(c2cc(C(F)(F)F)ncn2)=O)C(O)C1 78585,c1(C(=O)NCC2(F)CC(NC(=O)CC3CSCCS3)C2)ccc(F)c2ccoc12 78586,C1(C)(C(=O)NCC(C)(C)OCCNC(c2c(C)n(C)nn2)=O)CCC(=O)NC1 78587,c1(NC(C2C(C(=O)NC3CC4(CC4)C3)C2)=O)cccc(I)n1 78588,CCC(CC(=O)NCCc1ccccc1C)NC(=O)Cc1coc(C)n1 78589,N1(C(C(C(C)C)N2CCCCC2)=O)CC2CCC1CN2Cc1ccc(CF)cc1 78590,Cc1ccc2c(C(=O)NCC3CN(C(=O)CC(C)CC(C)(C)C)C3)cccc2c1 78591,S(=O)(=O)(c1ccc([N+](=O)[O-])cc1Cl)NCC1CCCN(C(C2(C)CCCC2)=O)C1 78592,C1(NC(c2c(C)scc2)=O)CC(O)CN(C(c2cc(Br)no2)=O)C1 78593,c1(C(N(CCCNC(C23CC(C2)C3)=O)CC)=O)cc(Br)cc2c1CCN2 78594,C1(F)(CNC(=O)CCSc2ccccn2)CCN(C(C2(O)CCCC2)=O)C1 78595,c1(C(=O)NC(CCNC(C(CCC)N(C)C)=O)C)cc([N+](=O)[O-])n(C)n1 78596,C12(CC(O)C1)C(=O)N2.CC1CC1C(=O)NCC(=O)NCCCO 78597,Cc1cc(C(=O)NC(CO)CCCCNC(=O)C(C)C(C)(C)C)cc(=O)n1C 78598,Cn1nnc2ccc(C(=O)NCC3CCC3NC(=O)C=Cc3cccnc3)nc12 78599,Cc1nc(CNC(=O)C(=O)NCc2ccccc2OC(C)C)ccc1F 78600,N1(C(c2cc(C(CC)CC)no2)=O)CC(C2CN(C(C3(CN(C)C)CC3)=O)C2)C1 78601,C1(CNC(=O)CCNC(=O)CC2OCCCO2)CC2CCC1CC2 78602,CC1(CO)CCCC1NC(C1CCC1NC(C1CC1(F)Cl)=O)=O 78603,N1(C(=O)Cc2ccc(Cl)cn2)CC2CCCN(C(C3COC4(CCC4)C3)=O)C2C1 78604,c1(CC)nc(N(C)CC2CCCN2C(=O)C(O)CC(C)(C)C)c2ccsc2n1 78605,C1(F)(C(=O)NCCC(C)CO)CCN(C(=O)C=Cc2cn(C)nn2)C1 78606,C(=O)(CCCCCF)N1C(C(C)NC(c2cc(OC)ns2)=O)CCCC1 78607,C(=O)(C1CCc2snnc21)N1CCC(NC(c2nn(C)c(C3CC3)c2)=O)C(O)C1 78608,c1(C(N2CCC(C)(NC(C=CCOC)=O)C2)=O)ccnc2ncsc12 78609,c1(NCC2(CC)CCOCC2)ncccc1S(=O)(=O)NC1(C(C)C)CCC1 78610,C1(CC(=O)N(CCC(C)NC(C=CSC)=O)C)CCCCN1C(=O)OC(C)(C)C 78611,c1(C(N2C3(CNC(COC)=O)CCC2CC3)=O)cccc2c1OC(C)C(=O)N2 78612,Cc1ccc(C(N2CC(NC(c3cncc(N)n3)=O)C(C(F)F)C2)=O)nc1C 78613,N1(C(c2ccc(CC)c(F)c2)=O)CCN(C(c2cccc(C)n2)=O)C(C)C1C 78614,C1(CNC(=O)CC2(C(F)(F)F)CC2)CCCN(C(=O)C(F)(F)c2cscn2)C1 78615,N1(C(c2c(C)nsc2)=O)CCCC2(C1)C(NC(c1cn(C)nc1Cl)=O)CCN2C 78616,N#Cc1ccc(C2(CN=c3[nH]nc(-c4ccccc4)s3)CCCC2)cc1 78617,N1(C(C(C(C)C)NC(C)=O)=O)CCN(C(=O)CNC(=O)C2CC2)CCC1C 78618,Cc1cc(C(=O)NC2CCCN(C(=O)CSC3CC3)CC2)ccc1[N+](=O)[O-] 78619,c1(C(N2CC(NC(C3CCN(C)C3=O)=O)C2)=O)ccc2c(O)n[nH]c2c1 78620,C1(CNC(CNC(CNC(C)=O)=O)=O)CN(C(c2cnncc2O)=O)CCO1 78621,C1(C(N(CC(C)NC(C2CCS(=O)(=O)CC2)=O)CC)=O)(OC)CCCCCCC1 78622,c12ccc(C)c(c1)N(C)C2=O.N1(C(C2C(C)(CC)C2)=O)CCC(NC(C)=O)CC1 78623,C1(C)(C(=O)NCCCNC(c2cc(-c3n(C)ccc3)[nH]n2)=O)CCCC(F)(F)C1 78624,c1(C(=O)NCCCC(C)NC(C2CC3(CC(=C)C3)C2)=O)ccc2sc(=N)[nH]c2c1 78625,C1(N(C(C(C)OCCOC)=O)C)CCC(NC(=O)CC2COCCN2C)CC1 78626,n1(C(C(=O)NCCN(C(c2c(C)snn2)=O)C)C)nc([N+](=O)[O-])cc1C 78627,c1(C(N(C2CCCC(NC(c3occc3F)=O)C2)C)=O)ccc(F)cn1 78628,Cc1nc(CNC(=O)C(O)CNC(C2CC(C3CC3)C2)=O)sc1C 78629,C1(CNC(CNC(CCC)=O)=O)C(C(N2CCC(CC(C)C)C2)=O)C1(C)C 78630,Cc1cc2ncc(C(=O)NCC=CCNC(c3ccc(Br)c(F)c3)=O)cn2n1 78631,CC(CC(=O)N1CC(NC(=O)Cc2cc(F)cc(Br)c2)C(O)C1)C(F)F 78632,N1(c2snc(COC)n2)CC(CNC(=O)Cc2cnn(C)c2)OC(C)(C)C1 78633,N1(C(C2(COC)C=CCC2)=O)C2CCC1CN(C(=O)CCCc1cncs1)CC2 78634,C1(C(N2C(C)C(NC(C3(C)CC3)=O)CC2)=O)CC2C(C1)C2(F)F 78635,CCC(C)(COC)C(=O)N1CCC(CNC(c2cnn(C3CCCC3)c2)=O)C1 78636,CCC(CC(C)C)C(=O)N1CC(O)(CNC(c2nc(Cl)sc2Cl)=O)C1 78637,c1(NC(N2CCCC(CCCO)C2)=O)cccc(-c2ccc[nH]2)c1 78638,c1(CC)cc(C(=O)NCC2CC(NC(C3CN(C(C)C)C3)=O)C2)oc1CC 78639,C(=O)(CCC1=CCCCC1)NCCCCCNC(c1nc(N)c(Br)cc1)=O 78640,CC1=NOC(CNC(=O)C(C)(C2CC2)N(C(=O)CN=[N+]=[N-])C)C1 78641,c1(C(=O)NCC(CC=C)NC(=O)Cc2cccnc2C)ccc([N+](=O)[O-])cc1O 78642,C1(C)(C(=O)NC(c2cn(Cc3cnc(C)nc3)nn2)C)Cc2ccccc2C1 78643,CCCC(CC)CCC(=O)NC1CC2(C(=O)NC(C)(CO)CO)COC1C2 78644,C12(NC(=O)OC(C)(C)C)CCCC1CCN2C(c1ccc(F)c(N)c1F)=O 78645,C(CNC(=O)CCC(C)N(C)C)(CC(F)(F)F)NC(Cn1c(C)nnn1)=O 78646,C1(C(=O)OCC)CC(C(N2CCC2(C)NC(CCC)=O)=O)C1(C)C 78647,C(C(CN=c1[nH]cnc(Cl)c1Br)CCCl)NC(c1ccc(NC(C)=O)cc1O)=O 78648,C1(N(CC(C)C)C(C2C(C)(CC)C2)=O)CCN(C(=O)CCC=CC(C)C)CC1 78649,C(CCC(=O)NCC1=NOC2CCCC12)(C(C)C)NC(c1nc(C)oc1C)=O 78650,N1(C(C(C)(C)C2CCC2)=O)CCOC2(CCN(C(C3CC(=O)N(O)C3)=O)CC2)C1 78651,c1(C(N2C3CN(C(C4N(CC)CCC4)=O)CC2C3)=O)cccc2c1ccn2C 78652,C1(C(=O)NC(CC)C(F)(F)F)CN(C(c2ccncc2F)=O)CC12CCC2 78653,CC1C(C(=O)NC2(C(F)(F)F)CC(F)C2)C(C(=O)O)C1(C)C 78654,c1(CC(=O)NC2CC(C(=O)NCc3c(C)nns3)OCC2)c(F)cccc1F 78655,C1(O)(CNC(c2cccc[n+]2[O-])=O)CCCN(C(=O)C(Cl)=CCl)CC1 78656,c1(OCCC(N2C(Cn3cc(CCS(C)(=O)=O)nn3)CC2)=O)ccc(F)c(F)c1 78657,c1(C(N(C2CN(C(c3cc(-c4ccco4)no3)=O)C2)C)=O)cn(CC2CC2)nn1 78658,Cc1cc(C(N2CCC(N(C(=O)CC3COC(=O)C3)C)C2)=O)ncc1CO 78659,N1(C(c2c(C)noc2C2CC2)=O)CC2CC1CN2C(=O)C(F)OC(F)(F)F 78660,C(C)(C(=O)NC1CC(OCC(=O)NCCc2ccncc2)C1)(C1(C)CC1)OC 78661,N1(C(c2c(C)cccc2Cl)=O)CC2(CCCC2NC(C2CCC3CC3CC2)=O)C1 78662,c1(COC)ccc(C(N2CC(O)(C(C)NC(=O)C(C)c3ncco3)C2)=O)s1 78663,CCC(CNC(=O)CCCN(C(=O)C(C)NC(C)(C)CC)C)CO 78664,CC1(C)CC(NC(c2cccc(O)n2)=O)CN1C(C1CCN(S(C)(=O)=O)C1)=O 78665,N1(C(CCN(C(C2CCC(C)(C)OC2)=O)CC)=O)CC(S(N)(=O)=O)C1 78666,c1(C(C(=O)NC(C)C)N(C(CC)C#N)C)csc(C(F)(F)F)n1 78667,c1(C(N2C(C(C)NC(CN3CC(C)(OC)C3)=O)CCC2)=O)ccc(N(C)C)cn1 78668,Cc1ccc(CN2CCCC2CCC(=O)N(C)Cc2ccccc2)c(Cl)c1 78669,c1(CNC2(CNC(=O)CC3(CO)CC3)CC2)nc2c(cc1Cl)C(=O)OC2 78670,C1(NC(C(CC)N(CC)CC)=O)CCN(C(=O)C2=CCCCCC2)CC12CCC2 78671,c1(C(=O)NC2CC3CN(C(C4(C)CCCC4)=O)C(C2)C3)cccc2cccnc12 78672,C1(N(C(C(=O)N(CCN(C(C=C(COC)C)=O)C)C)C)C)CCCOC1 78673,C=CCCCCC(=O)N(C)CC1(C)CCCC1NC(c1ccc(C)s1)=O 78674,C1(OCC(=O)N(C)CC2(NC(CN(C(=O)OC(C)(C)C)CC)=O)CC2)CCCCC1 78675,N1(C(Cc2ccn(C(C)C)n2)=O)CCCN(C(=O)CO)C(C)C1 78676,c1(OC)ccn2c(C(=O)NC(C)C(C)NC(=O)CSc3nncn3C)cnc2c1 78677,CN=C(NCc1cc(-c2ccccc2)n[nH]1)NCC(Br)=C(C)C 78678,N1(C(C2(CC)CC2(F)F)=O)CC2C(CNC(=O)CC3CCCC3)C2C1 78679,Cc1ccc2c(=NC(=O)C3CCCCN3C(C3CCC(C)O3)=O)[nH][nH]c2n1 78680,C(=O)(C(COC)CC(C)C)NCC(=O)NC(COC)C(=O)OC1CCC(OC)CC1 78681,C=CC1(CO)CCN(C(=O)C(CCC)NC(=O)CSCC(N)=O)C1 78682,C1(NC(c2cc(C(F)F)ccn2)=O)CC2(CCCCN2C(C2(C(F)F)CC2)=O)C1 78683,C(=O)(CC(O)C(=O)NCCC12CCC1CN(C(C1CCC1)=O)C2)OC(C)(C)C 78684,S(=O)(=O)(c1cccc(=NCc2cn(C)nn2)[nH]1)NC(c1ccn(C)n1)CO 78685,N1(C(C)=O)CC(O)CC1C(=O)NCC1CCN(C(C2(C)CSC2)=O)C1 78686,C(=O)(CCCCCCCCCO)N(CC(CC)NC(C1(Cl)CC1(F)F)=O)C 78687,Cc1ccccc1C=CC(=O)NC(C(=O)NCC12CCN(CC1)C2)c1cccs1 78688,c1(C(C)C#N)cccc(C(N2CC(O)CC2C(=O)NC2CN(c3nncs3)C2)=O)c1 78689,c1(C(C(=O)NCC2CCCC2)NC)cc(C(C)(C)C)oc1C.C1(C)C2CCCC12 78690,N1(C(C(COC)C)=O)CCCC2(C1)CN(C(c1nn(C)c(C)c1Cl)=O)CCO2 78691,n1(CC)cnc2c(N(CC(C)CO)C)nc(N3CCC4(CCCOC4)C3)nc12 78692,C1(N(C(C(C)SCC)=O)C)CCCN(C(=O)CCc2nc(CC)no2)CC1 78693,c1(C(=O)NCC(C)CN(C)C(C2CNC(=O)N2C)=O)coc2c(F)cc(F)cc12 78694,O=C(CCCC1CCCC1)N1CCC(CNC(C2(n3cnnn3)CC2)=O)C1 78695,C1(C(=O)NC2(CC=C)CN(C(=O)C(C)NC(c3ccoc3)=O)C2)CCNC(=O)C1 78696,c1(OC)ccc(=NC(=O)C23CC2CN(C(c2cc(Br)ncc2F)=O)C3)[nH]n1 78697,n1(CC(=O)N(C2CN(C(c3cnn(C)n3)=O)CC2(C)C)C)nc(Cl)ccc1=O 78698,N1(C(C23C(C)OC(C)(C2)C3)=O)CCCN(C(=O)C(F)F)CC1C 78699,N1(C(C(C)SC(F)(F)F)=O)CC2CC1C2CNC(C1(CF)CC1(F)F)=O 78700,c1(C(N2CCC(NC(C(C)C3CC3)=O)C(F)C2)=O)c(O)cnc2ccccc12 78701,C1(CNC(C=CC=CC)=O)(OC)CCC(C)C1.C12(F)CN(C1)C2=O 78702,N1(C(C(C)C2CCCO2)=O)CC2(NC(c3ccc(Br)cc3N)=O)CCC1CC2 78703,C1(CNC(=O)C(=O)NC2CC2)CCC2CN(C(c3ccc(O)cc3)=O)CCC2C1 78704,C1(NC(C(C)(C)SC)=O)CC12CCN(C(=O)Cc1ccoc1C)CC2 78705,C(c1cn(C)cn1)=C(C(=O)NC(CNC(C(C)OCCN(C)C)=O)C)F 78706,C(=O)(C(C)N(C(C1CCC1C)=O)C1CC1)NCCN(C(C)C)CC 78707,c1(C(N(CC(CNC(c2n(C(C)C)ccc2)=O)C)C)=O)[nH]ncc1C#N 78708,CCCCS(=O)(=O)NCC(=O)NC1CC(NC(=O)CCCCSC)CC1O 78709,c1(C(C(=O)NCCC(C)NC(C2(Cl)CC2)=O)NC(C)=O)ccccc1 78710,c1(C(=O)NC(CCCNC(c2nnc(C)s2)=O)C)cccc(CO)c1C 78711,C=CCCN=C(NCC(CC)n1cccn1)NC1CCC(CC)CC1 78712,c1(C(C(N2CC(NC(C3(OC)CCCC3)=O)C2)=O)N(C)C)c(F)cccc1F 78713,N1(C(Cc2ccc(OC)nc2)=O)CCC2C(C1)NC(=O)CN2C(=O)CSC1CC1 78714,N1(C(C(CC)(F)F)=O)Cc2occ(C(N3CC(CO)CC3CO)=O)c2C1 78715,Cc1cc(C)n(CCNC(=O)CC(N)Cc2ccc(F)cc2)n1 78716,Cc1sc(Br)nc1C(=O)NCC1(C)CCN(C(C2CC(F)(F)C2)=O)C1 78717,c1(C(C(=O)NC2C(OC)CN(C(C3CN(C)C3)=O)C2)O)ccc(Cl)cc1Cl 78718,Cc1cc(C)c2c(=NC(=O)NC(c3ccnc(Cl)c3)C)[nH]sc2n1 78719,Cc1nc2ccc(S(=O)(=O)NC3CCC4CCCCC4C3)cc2o1 78720,Nc1ccc(Br)c(F)c1CNC(c1ccccc1)C1CC1 78721,N1(C(c2cn(CC)nn2)=O)CC2CCC2(CNC(c2oncc2C)=O)C1 78722,c1(CCC(=O)NCC2N(C(C(CC)C(C)C)=O)CC2)ccccc1[N+](=O)[O-] 78723,C1(N(C(C(CC)F)=O)C)CN(C(c2ccc(C(=O)NC(C)C)cc2)=O)CC1(C)C 78724,C1(=CC(=O)NCC2COCC2NC(C2CCOC2)=O)C2CC3CC(C2)CC1C3 78725,N1(C(c2nc(CC)oc2)=O)CC(NC(c2sc3cncn3c2C)=O)C(C2CC2)C1 78726,C(CCCCCC(=O)N1CC2CCC2(CNC(=O)C(O)C(C)(C)C)C1)SC 78727,C(=O)(CC(C)(C)C(F)F)N1C(CNC(C(CCC)CC)=O)CCC1 78728,c1(C(=O)NCC(C)CNC(=O)CCCC(C)(C)C)n[nH]c2c1CCCCC2 78729,Cc1cc(C(=O)NCC(C)(C2CC2)NC(c2ccn(C)n2)=O)sc1C 78730,C(N=c1[nH]c(=NC(CCO)c2ccco2)[nH]c2ccsc12)C1(S(N)(=O)=O)CC1 78731,c1(NC(c2occ(C(C)=O)c2)=O)ccc(NC(C2(O)CCCCCC2)=O)cc1C 78732,C1(N=c2[nH]nc(C(F)F)s2)(NC(C2(C)CCC(C)(C(=O)OC(C)(C)C)C2)=O)CC1 78733,C(=O)(N=c1cc(C)n(C)[nH]1)C1OCCC(NC(CCCOCC=C)=O)C1 78734,N1(C(CC)=O)CCCC1C1(NC(C2CC(C)(CC)C2)=O)CC1 78735,c1(OCCOC)ccc(C(=O)NC2CCC(NC(=O)C(C)C(C)C)CC2)cc1 78736,C1(C(=O)NCC2CN(C(C3C(OCC)C3)=O)CC2C)CCc2cncn2C1 78737,N1(C(COCC(C)C)=O)CC2C3CCC(C2C1)N(C(c1ncccc1CO)=O)C3 78738,Cc1cccc(C(=O)OCC(=O)NC2CC2CNC(c2nn(C)cc2C)=O)c1 78739,C1(NC(c2n(CCOC)nnn2)c2ccncc2)CCc2ncccc2C1 78740,c1(CC)ccc(CNC(=O)C(CCSC)NC(=O)C2=CCSC2)cc1 78741,Cc1nnc2n1CCC2(C)C(=O)N1CCC(C)(NC(=O)CC2COCCOC2)C1 78742,CCCC(C)C(=O)N1CC=CC1(C(=O)NC1CC(C)(C)C1)COC 78743,C(=O)(C1=NOC2(CCN(C(c3c(OC)cccc3)=O)C2)C1)NC1CC2CCC1O2 78744,Cc1nn(C)c(C)c1C.N12CC(C1)CN2C(=O)CN(C)C.C(C(C)C)S 78745,N#CC1CCCCC1NC(C1CCN(C(=O)CCCC#N)CC1O)=O 78746,c1(N2CCC(CC=C)C2)cc(NCC(C)CC(C)C)nc(C(F)(F)F)n1 78747,CC1CC=C(C(=O)NC2COCC2NC(c2cccc3nccn23)=O)CC1 78748,C1(C)(CCC(=O)NC(C#C)(C)C)CCN(C(c2csc(C#N)c2)=O)CC1 78749,CC1(C)CCCC(C(=O)NCCC2CN(C(c3cncc(CO)c3)=O)C2)O1 78750,c1(OC)cc(C)c(Cl)cc1S(=O)(=O)N1CCN(C(c2cnc[nH]2)=O)C(C)C1 78751,CC1=C(C(=O)NCC2(NC(=O)CC3CCCN3C(C)C)CCOCC2)CCO1 78752,Cc1c(C(=O)N(CCC(C(C)C)NC(C2CSC2)=O)C)[nH]c2c1CCCC2 78753,c1(CCOC)cccc(CN2CCNC(COC(C)(C)C)C2)c1 78754,N1(C(C2CC(N(C(C(C)n3ccnc3)=O)C)C2)=O)CC2CC1CN2C(C)C 78755,C=CC1(CC(=O)NC(C)C(C)NC(=O)CC2CSC2)CCCCC1 78756,C1(NC(C(CCOC)OC)=O)CCN(C(=O)Cn2nnnc2C(C)C)C(C)C1 78757,N1(C(c2ccc(CCC)s2)=O)CCC2(CC(NC(C3(C(=O)NC)CC3)=O)CO2)C1 78758,N1(C(COC(C)C)=O)CCC(C)(C)C(NC(=O)COCC2(F)CC2)C1 78759,C1(NC(C2CC(=O)NC2)=O)(CO)CCN(C(c2ncccc2OCCF)=O)C1 78760,c1(C(=O)NC(CC)CNC(C2(F)CCOC2C)=O)c(C)nn(CC)c1C 78761,Cn1cnc(CCNC(=O)C(C2CC2)N(C(=O)CSCC(N)=O)CC2CC2)n1 78762,CCC(C(=O)N1CC(OCC(=O)NC2CCOC2)C1)OC 78763,N1(C=O)CCN(c2ccc(-c3sccc3C)cn2)CC1.Cc1nc(C=O)co1 78764,CC1(C)COCCC1C(N1CCC(CC(N)=O)(NC(C2(CO)CCC2)=O)CC1)=O 78765,C(CCC(F)(F)F)N(C(c1scc(C(C)=O)n1)=O)C 78766,C(=O)(CC(CC)C(C)(C)C)NCC(CC=C)NC(=O)CNS(=O)(=O)C1CC1 78767,c1(C(N(CC(C)NC(c2cc3ccnn3cn2)=O)C)=O)c(F)ccc(N)c1F 78768,c1(-n2c(CCC=C(C)C)nc(Cc3ccncc3)n2)cccc2nc[nH]c12 78769,C(=O)(CC(C)(C)CNC(=O)Nc1cc(C(C)(C)C)ccn1)OCC 78770,C1(C(=O)NC(C(NOCC(=C)Cl)=O)c2ccnn2C)CC2(CCC2O)C1 78771,CC(CCCC(=O)NCC(C)C(C)O)NC(=O)CC=Cc1ccccc1 78772,c1(CC2N(C(c3sccc3Cl)C(=O)NC)CCC2)ccc(OC)cc1 78773,c1(C(N(CCC)CCNC(C2CCC3CC3CC2)=O)=O)ccc2n[nH]cc2c1F 78774,c1(C(=O)NC(C)C(=O)NC2CC(CNC(=O)CCCF)C2)ccc([N+](=O)[O-])cc1 78775,C#CC1(O)CCN(C(C)C(=O)NC(C)CCCCNC(C2CCC(F)C2)=O)CC1 78776,CCCCCCCCCC(=O)N1CC(NC(=O)CC(C)(C)C(F)(F)F)CC1C 78777,C1(CC(=O)NCCCCCNC(C2(SC)CCC2)=O)CCCS1(=O)=O 78778,c1(C(=O)NCC(n2cncn2)C)ccn(CCNC(=O)CCCc2ncco2)c1 78779,C1(C(=O)NC(C2(C(=O)NCC(C)(C)C)CC2)C)CCC2(CC2)C1 78780,N1(C(c2cc(C)c(Br)o2)=O)CC(NC(c2snnc2C)=O)CC(F)C1 78781,C(=O)(CCS(N)(=O)=O)NCC(N1CCC(C)(CO)C1)=O.C1CN1CCO 78782,c1(CN2CC(C)(CNC(c3cccc(OC)c3)=O)C2)cc([N+](=O)[O-])ccc1Cl 78783,C1(NC(=O)CC2COCC2O)C2CN(C(=O)CCCc3ccccn3)CC12 78784,C1(NC(=O)CNC(=O)C2CC2)CC2CCC1(C(=O)NCC1(F)CCC1)C2 78785,C1(N2C(=O)C2)CCN(C(C2CCOC2C(F)(F)F)=O)C1.C(C(C)C)SC 78786,C1(NC(C2(c3nc(C)on3)CC2)=O)CCCN1C=O.C12C=CC(C1)NC(=O)C2 78787,C1(CNC(CC2C(C)CCO2)=O)CCCCCN1C(c1csc(=N)[nH]1)=O 78788,N1(C(Cc2c(C)occ2)=O)CCOC(CCNC(=O)CC2COCCOC2)C1 78789,Cc1ccc(F)c(C(=O)NC(C2(O)CCN(C(=O)CCC3(O)CCC3)C2)C)c1F 78790,C1(C)(C(=O)NC(C2CCOCC2)CC)CCN(C(c2cc(CO)[nH]n2)=O)CC1 78791,C12(NC(c3snnc3C3CC3)=O)CCCC1CN(C(=O)Cc1ccsn1)C2 78792,C1(C(N2CCC(C(C(=O)NCCc3ccc(O)cc3)F)C2)=O)CCC2(CCC2)C1 78793,c1(C(N2CC(CC)N(C(C3CC4CC4C3)=O)CC2)=O)ccc2[nH]ccc2n1 78794,C1(CNC(c2c(C)sc(C)c2Br)c2n(CCC)nnn2)CSc2ccccc2O1 78795,N1(C(C(=O)N(CC)CC)=O)CC2C(NC(=O)CCC3CCCCO3)C2C1 78796,CCC(CC)(C(C)C)NC(c1cc(CCNC(=O)C(C)=CC(C)(C)C)on1)=O 78797,c1(C(C)NC(CONC(Cc2scc(C)c2)=O)=O)ccc(F)cc1 78798,N1(C(c2c(C)[nH]cc2)=O)CC2C3CCC(C2C1)N(C(C1CC(C)CO1)=O)C3 78799,C1(CC)CC(N=c2[nH]c3c(c(=NCC(F)C4CCCCC4)[nH]2)SCC3)C1 78800,c1(OC)cc(F)c(C(N2CC(O)C(O)C2CNC(=O)C(O)CSC)=O)cc1OC 78801,C1(C(=O)NC2CN(C(C(C)OCCOC)=O)C2)CC2(CCCCC2)S1(=O)=O 78802,c1(C(=O)NC(C)(C)CNC(C2(C)CCCOC2)=O)cc2c(nn1)CCCC2 78803,N1(CC)CCC(O)C(N=c2ncnc(NC)[nH]2)C1 78804,c1(C(=O)NC2CN(C(C3C(C)CC(=O)N3)=O)C2)nnc(O)cc1O 78805,C(C)(C(C(=O)N(C1(CCO)CC1)C)C(C)C)NC(C(C(=O)OC)C)=O 78806,c1(C(=O)OCC)cc([N+](=O)[O-])cc(CNC2CCCN(C(C)(C)C)C2)c1O 78807,C1(NC(COc2cccc(OCC)c2)=O)CCN(C(=O)CC2CC2)CC12CCC2 78808,c1(C(N2CC(CN(C(=O)C(C)(O)C3CC3)C)C2)=O)cc2n(n1)CCCO2 78809,N#CC1(C(N2CC(NC(=O)C(N)=O)C(n3cccn3)C2)=O)CCSCC1 78810,Cc1onc(C2CCCCC2)c1C(=O)NCC1(NC(=O)CC(F)(F)F)CC1 78811,Cc1ccc(F)c(C(=O)NCC2(C)CC(NC(c3cnc4n3CCS4)=O)C2)c1F 78812,N1(C(C=CC2(C)COC2)=O)CC(C(=O)NCC2C3CCCCCC23)C(C)(C)C1 78813,CC(C)(CC(F)(F)F)NC(C1C2CCC(C2)C1N)=O 78814,c1(C(=O)NC2CCc3nccn3C2)cccc2cc(Cl)ccc12 78815,C1(CC)CNC(=O)CN1C(C1(NC(C2CCCCNC2=O)=O)CCCC1)=O 78816,C1(N(C(c2nn(C)nc2Br)C(=O)NCC(F)F)C)CS(=O)(=O)C12CCOCC2 78817,C1(C(=O)NC2CCC(CNC(CCC3C(C)(C)C3)=O)C2)CCc2n[nH]cc2C1 78818,c1(C(=O)NCC(CC)NC(C2(CC)CC(F)(F)C2)=O)cnc(S)n1C 78819,N#CC1(CNC(C2CCN2C(C2CC2(Cl)Cl)=O)=O)CCC1 78820,CCCC(O)C(=O)NCCCN(C(C1C2CC2C2CC12)=O)Cc1ccccc1 78821,C1(NC(COCC#C)=O)(CNC(CC2(OC)CC2)=O)CCCC1 78822,c1(SCC(=O)NCC2CCCN2C(c2ncccc2Cl)=O)ccsc1[N+](=O)[O-] 78823,CC(CNC(=O)CC1CC1)CC(=O)NC(C)(CO)C1CC1 78824,CN=c1[nH]c(=NCc2cncc(C)c2)[nH]c(=NC2CCN(CCOC)C2)[nH]1 78825,Cc1cnc(C(=O)NCC2(CNC(=O)C(c3ccn(C)c3)C)CC2)cn1 78826,C1C(F)(F)C(=O)N1C.O(NC(=O)COC)CC(=O)OCC 78827,N1(C(c2ccc(Cl)cc2F)=O)CC2CCN(Cc3ccccc3[N+](=O)[O-])CC2C1 78828,C1(CNC(C=CSC)=O)CCC(C)(C)CN1C(c1sc(C)nc1C)=O 78829,C1(c2nc(C)on2)CCCN1N(C)Cc1cccc(C(F)(F)F)c1 78830,C1(NC(CS(=O)(=O)NCC)=O)(CNC(c2ccoc2C)=O)Cc2ccccc2C1 78831,C12(C(N3CCC(OCCNC(CCCOCC)=O)C3)=O)CCCC1CC(=O)C2 78832,c1(CNC2C(C(=O)NCc3ccc(C)cc3C)C2)cc(F)c(F)cc1O 78833,c1(C(N2C(CNC(C(CC)C)=O)CC(C)(C)C2)=O)ccc(S(N)(=O)=O)cc1F 78834,c12ccc(c(OC)c1)NC2.C1C(=O)N(C(C)C)N1CC.S(C)(=O)(=O)NC 78835,CC1CCNCC1NC(=O)C(=O)NC(c1cccc(F)c1)c1ccccn1 78836,N1(C(C(=CC2CCCC2)C)=O)CCC2(C=C(C(=O)N3CCOCC3C(N)=O)C2)C1 78837,c1(C(C(N2CC(COC)(NC(c3nccnc3N)=O)C2)=O)O)ccc(F)c(Cl)c1 78838,C(CC(C)(C)CNC(=O)C(=O)NCc1ncc(C)o1)OC 78839,C(=O)(CC(C)C(C)(C)NC(C1CC(C)N(C)C1)=O)N(CC(C(C)C)C)C 78840,CC1CC2(CCCC2)CN1C(C1CCC(C2CC2)N1C(C1CCCN1C1CC1)=O)=O 78841,CC1CC(NC(=O)C(c2cc(F)ccc2F)=O)CC(C)(C)C1 78842,N1(C(C(C)(C)c2ccccn2)=O)CCN(C(=O)C(O)CN2CCOCC2)CC1 78843,C(CS(=O)(=O)Cc1cn(C2COCC2CN)nn1)NC(CNc1onc(C)n1)=O 78844,C(C(C)C(F)C(=O)N(C)CCc1cccs1)NC(CCn1ncc(C)c1)=O 78845,C(=O)(C#CC1CCCCC1)NCC(c1cc(F)cc(F)c1)C 78846,c1(NC(C2(C)C(C)CN(C(C(CC=C)C)=O)C2)=O)ccccc1C(=C)C 78847,C(=O)(CCCCC(C)=O)N1C(C)CC(C(N2CC(C(CC)C)C2)=O)C1 78848,N1(C(C=C(C)C2CC2)=O)CCCC(N=[N+]=[N-])C1.C12CC(C1)OCC(=O)N2 78849,c1(C(=O)NCC(CNC(=O)CCOC(C)C)OC)c(C)cc(Cl)cc1C 78850,C(CCC(=O)N1CC(CC2CCCC2)C1)N(C(C(C)=C(C)C)=O)C 78851,CC1CN(C(c2ocnc2C2CC2)=O)CC(C)C1NC(=O)Cn1ccnn1 78852,Cc1nn(C)cc1C(=O)NC1CN(C(c2ccc(OC(C)(C)C)nc2)=O)C1 78853,Cc1ncc(C(C)NC(c2cn(CCNC(=O)CC34CCCC3C4)cn2)=O)s1 78854,c1(C(=O)NC2CCN(C(c3ccnnc3S)=O)C2)cc(N2CCCC2)ccn1 78855,CCC(C)C(=O)NCC(=O)N(C(C)CCNC(=O)Cc1cc(C)no1)C 78856,N1(C(c2c(OC)ccnc2)=O)CC(N=[N+]=[N-])CC1C(=O)NCCCCCO 78857,Cc1cc(NC(C2(NC(C3CC3(Cl)Cl)=O)CCSC2)=O)cc(CO)c1 78858,N1(CC(C)(C)NC(C(C)=C(C)C)=O)CCN(C(=O)C(C)(C)N(C)C)CC1 78859,N1(CC(=O)NC(C2(O)CCN(C(c3cn(CCO)nn3)=O)C2)C)CCNC(=O)C1 78860,c1(N(C)Cc2nnc(C)s2)nc(N2CCn3cc(Br)cc3C2)c2c(n1)CSC2 78861,C1(NC(CC2N(C(c3c(OC)cnnc3)=O)CC(O)C2)=O)CCN(C)CC1C#N 78862,N1(C(C(C)C(=O)N2CCOCC2)=O)CC2CCCC1(CNC(=O)C1CC1)C2 78863,C1(F)(CNC(C(=O)N(C)C)=O)CCN(C(=O)C(c2ccc(O)cc2)(C)C)CC1 78864,CC1(C)CC(NC(=O)C=Cc2cncs2)CN(C(=O)COC(F)(F)F)C1 78865,Cc1cnc(CNC(=O)COCCNC(=O)CN2CCCC2=O)[nH]1 78866,Cc1cc(C(=O)NC2C3CN(C(c4cc(F)cc(Br)c4F)=O)CC23)c(Br)cc1F 78867,c1(C(=O)NC2CC3CN(C(CSC(C)C)=O)C(C2)C3)nc2cc(O)ccc2[nH]1 78868,C1(CCC)COCCN1C(=O)CC(C1CC1)NC(C1OC2CCC1C2)=O 78869,N1(C(C2C(C=C)OCCC2)=O)CC2OCCN(C(c3oc(CC)cc3C)=O)C2C1 78870,Cc1csc2cc(C(=O)NCC(C)NC(c3csc4nccn34)=O)[nH]c12 78871,CC1(C)C(NC(=O)CCn2cnccc2=O)CCN1C(=O)CCn1ccnc1 78872,c1(C(=O)NC2CC(F)(CNC(CC(CC)SC)=O)C2)ccc2c(c1)CC(C)O2 78873,C#Cc1cccc(C(N2CCN(C(c3c[nH]nc3C(=O)O)=O)CC2)=O)c1 78874,c1(C(=O)NC23CC(NC(C4C(C)(CC)C4)=O)(C2)C3)cnc2ncc(Cl)cn12 78875,C1(C(N2CCC(N3CCC3)CC2)=O)CC(F)CN(Cc2ccc(C(F)(F)F)[nH]2)C1 78876,c1(C(N(CCCNC(c2c(OC)cco2)=O)C(C)C)=O)ncc(N)cc1C 78877,c1(OCC)cc(CNCCS(N)(=O)=O)ccc1OC(C1CC1N)=O 78878,C1(O)(CNC(C2(CCC)CC2)=O)CCCN(C(C23CCC(C)(C2)OC3)=O)C1 78879,C(=O)(CCCC(F)(F)F)NC(C1(O)CCN(C(C2CC(C)CC(C)C2)=O)CC1)C 78880,N1(C(CC2CCC(C)CO2)=O)CC(NC(c2nccc(C(F)F)n2)=O)CC(F)C1 78881,CCC(O)C(C)C(=O)N1CCC(CC)(NC(=O)CSc2nncn2C)CC1 78882,c1(CN2C(C(=O)Nc3ccc(Cl)nc3I)CC2)cc(F)ccc1[N+](=O)[O-] 78883,c1(CC)cc(=NC(=O)C(C)C(C)NC(=O)C(C)OC(C)=O)[nH]n1C 78884,CC1(C)C2CCC(C(=O)NC3C4CN(C(c5ccc(C(F)F)nc5)=O)CC34)C1C2 78885,C1(c2scc(C(=O)OC)n2)CN(N2CCCC(c3ccccc3F)C2)CCO1 78886,Cc1ncc2n1CC(C(N1CCCC(C)(C)C1CO)=O)CC2 78887,C(=O)(CCCCC(F)(F)F)N(C(CNC(c1nnc2n1CCCC2)=O)C1CC1)C 78888,CC1CCCCC1(CNC(C1C2(CC2)C12CC2)=O)NC(=O)CN1CC=CC1 78889,C1(C(=O)NC(c2cnn[nH]2)C)COCCN(C(c2ocnc2C(F)F)=O)C1 78890,c1(C(=O)NC23CCN(C(CCCSC)=O)C2CCC3)ccc2nc(C)cn2c1 78891,CC1=CCC(C(=O)NCC(C)(C)NC(C2CCCN(C(=O)OC(C)(C)C)C2)=O)CC1 78892,N1(C(C2(C)N(C(Cn3c(C)ncc3)=O)CC2)=O)Cc2ccc(Cl)nc2C1 78893,N1(C(C2C(=C)C2C(=O)OC)=O)CC2CN(C(c3cnn4ccsc34)=O)CC(C1)O2 78894,C1(C(=O)NCCCNC(c2ccc(OC(C)C)cn2)=O)CC2(C1)CC2(F)F 78895,c1(C(n2cc(C(C)N(C(=O)CCc3ccsc3)C)nn2)C)cccc(Cl)c1Cl 78896,C(=O)(C(CN(C(CCO)C(F)F)C)Cc1ccc(OC)cc1)NCCCOCC 78897,Cc1c(N)cc(C(N2CCC(CCNC(=O)C(C)CC(C)(C)C)CC2)=O)cc1N 78898,Cc1cc(NC(c2ccccc2O)=O)sc1C(=O)NC1CONC1=O 78899,C1(NC(C(CC)N2CCCC2=O)=O)CN(C(=O)CN(C(=O)COC)C)CCC1F 78900,C(=O)(C(C)CN(C)C)NC(C1CCCCC1)C(=O)NC(C)COC(F)(F)F 78901,C1(CC)CN(C(=O)CCc2c(C)noc2C)CCN1Cc1ccccc1OC 78902,C(c1ccc(Br)cc1)=CCC(=O)NCC(CNC(C(C)C1CC1)=O)CO 78903,N1(C(C(CCCC)O)=O)CC2CCCC2(CNC(c2ncc(C)cc2OC)=O)C1 78904,C1(NC(c2c(CC)n(C)nn2)=O)CCCCCC1NC(=O)CCCn1ccnn1 78905,N1(C(C2N(CC)CCOC2)=O)CCCC(NC(=O)C=Cc2cccc(F)c2)CC1 78906,c1(C(=O)NC(C(=O)NCCN(CCCC)C)CC(F)F)c[nH]c2ccccc12 78907,C(C)(CCCNC(=O)NC1CC(N2CCOCC2)C1)(OC)OC 78908,C1(CC)(CNC(c2cc(I)cs2)c2nnnn2C)CCCO1 78909,CC(C)C(N=[N+]=[N-])C(=O)NC(C)(C)C(=O)NC1CC(CO)C12CCC2 78910,C1(NC(C(C)(C)F)=O)CC2(C1)CN(C(C1(Cc3cnn[nH]3)CCCC1)=O)C2 78911,C1(C(=O)NC2C3CN(C(C=CC(C)C)=O)C(C3)CC2)CC2CCC(C1)S2(=O)=O 78912,Cc1ncc(NC(C2CCN2C(c2cc(Br)cnc2F)=O)=O)c(C)n1 78913,C1(O)(C(C)NC(c2nc(C(C)OC)oc2)=O)CCN(C(=O)C2=COCCC2)CC1 78914,C1(C(=O)NC(C2CCN(C(c3csc(O)n3)=O)CC2)(C)C)CC1C1CC(F)(F)C1 78915,C(=O)(C(F)C(C)CNC(=O)C(C)OCC=C)NCCSCC#C 78916,c1(C(C)C)ccc(C(N2CC(NC(=O)CC(C)c3cccnc3)C(O)C2)=O)nc1 78917,N1(C(c2c(C)snn2)=O)CC2ON=C(CNC(=O)CNC(=O)OC(C)(C)C)C2C1 78918,c1(NC(c2n(CC(=C)C)nnn2)c2cnc(C(C)(C)C)[nH]2)cc(C)cnc1OC 78919,C1(C(=O)NC(c2cnoc2)C2CC2)CCN(C(=O)CCc2ccccc2)CC1O 78920,C1(C(=O)NC(c2cnn(C)c2)CC)CC2(CCN1C(C1CC(=O)C1(C)C)=O)CC2 78921,Cc1nn(C)c(C(=O)NC(C)CCC2CCCC2)c1I 78922,C1(C(C)C)CN(C(=O)Cc2cn[nH]c2)CCN1C(c1cc(Cl)n(C)n1)=O 78923,c1(C(=O)CN2CCCC2c2cn(CCn3cccn3)nn2)c[nH]c2ncccc12 78924,c1(CN2C(C(=O)Nc3cnn(C(F)F)c3)CC3CC32)cc(Cl)c(Cl)c(Cl)c1 78925,N1(C(C(CC)C2CCOCC2)=O)CCN(C(C2(C)COC2)=O)C(C)C1 78926,c1(-c2ccn(C(C)C)n2)n[nH]c2cccc(C(=O)Nc3ncc(F)cc3F)c12 78927,CCC1=NOC(C(=O)NC(C2CCCN2C(=O)C2CC2)(C)C)C1 78928,Cc1cc(C(=O)NC(c2ccc(N(C)C)cc2)CNC(=O)C(C)O)ncn1 78929,N1(C(CC2CCC(C)(C)C2)=O)CCN(C(C2(C#N)CC23CCC3)=O)CC2(CC2)C1 78930,CC(C)CCC(C(=O)O)NC(c1ccc(F)nc1)=O 78931,O=C(O)CC(C(=O)NC1CCC(c2nc[nH]n2)CC1)C1CC1 78932,C(=O)(CC(C(F)F)NC(C1CCC1C(C)(C)C)=O)NCCC[Si](C)(C)C 78933,O=C1CCC2(CCCN(C(c3cccc4oc(O)nc34)=O)C2)CN1 78934,c1(C(C(=O)N(CCCNC(CC=C=C)=O)CC)N(CC)CC)cccc(Cl)c1 78935,C1(C(N2CC(NC(=O)CC(O)CC3CC3)C(O)C2)=O)Cc2ccccc2O1 78936,CC1CN(C(C2C3CCCC3CN2C(=O)CS(C)(=O)=O)=O)C(C)C(C)(C)O1 78937,C1(CC(=O)N(CCC(F)(F)F)C2(C(=O)OC)CCC2)CN(CC)CCC1C 78938,C12(CNC(c3ccccc3)C(=O)NCCC#C)CCC(CC1)C2 78939,C(C(N=[N+]=[N-])C(=O)NCC1CCCN(C(=O)CCN2CCN(C)CC2)C1)OCC 78940,c1(C(C(=O)N(CCNC(C2CC3(CC3)C2)=O)C2CC2)(F)F)cccc(F)c1F 78941,Cc1cc(C)c(NC(=O)C(C(C)(C)C)n2ccnn2)cc1O 78942,C1(OC)(OC)CC(C2CCN(c3nnc(-c4ncccc4F)n3CCC#N)C2)C1 78943,c1(C(N2CCCC2)=O)ccc(-c2ncno2)cc1.CCCN 78944,Cn1[nH]c(=NC(=O)C2(C)CN(S(=O)(=O)CCCCCl)C2)c2ccc(Br)cc12 78945,C1(CNC(CCCCC=CC)=O)CN(C(=O)C=C(Cl)Cl)CCC12CCC2 78946,N1(C(c2c(C)n(C3CC3)cc2)=O)CCC(C2CCN(C(=O)CSS(C)(=O)=O)C2)C1 78947,O=C(CC1=CCOCC1)N1CC(C2(NC(C3CCCC4(CCC4)C3)=O)CC2)C1 78948,C1(ONCC=C2CC(=C)C2)COC2(CCN(C(C(C)(C)C)=O)CC2)C1 78949,C12(C(N(CC(CC)O)CC)=O)COCC1CN(C(=O)CCc1ccncc1)C2 78950,C1(C(=O)NCC(C2CC2)NC(c2snnc2C2CC2)=O)CC2CC1C1C2C1(F)F 78951,N1(C(CN(C)C)=O)CCN(C(C2CCCC2(F)F)=O)CC(C)(C)C1 78952,N1(C(=O)Nc2c(OC)ccc(-c3cnco3)c2)CC(F)(CO)C2(CCC2)C1 78953,c1(CC)cccc(C(=O)NCC(C)(C)NC(c2cc(C3CC3C)on2)=O)c1 78954,CC1CC(C)CN(C(=O)C(N2CCCC2c2ccccc2)=O)C1 78955,CN(C)NC(=O)CCC(=O)NC1CC2(C(=O)NC3CC3(C)C(F)F)COC1C2 78956,N1(C(CCc2ccc(C)cc2)=O)CCN(C(=O)C(C)c2ccsc2)C2CC12 78957,N1(C(C(C2CCC2)OC)C(=O)NC(C)C)CCn2c(CCO)nnc2C1 78958,C1(CNC(C2CCC(C)O2)=O)C2CN(C(=O)CCNC(N)=O)CC12 78959,C1(CNC(C(C)NC(C)=O)=O)CC2COCC2N1C(c1cncn1C(C)C)=O 78960,c1(C(=O)NC2CN(C(C(C)CN(C)C)=O)CC2C2CC2)cc2cc(F)ccc2[nH]1 78961,N1(C(C2(CC)CCC2)=O)CCC2(CCN(c3ccc(C#N)nc3)C2)C1 78962,c1(C(=O)OC)cc(S(=O)(=O)N(C)Cc2ccc(C(=O)Nc3cc[nH]n3)cc2)cs1 78963,N1(C(C2(C(=O)OCC)C=CCC2)=O)CCN(C(=O)CNc2ncccn2)CC1 78964,N1(C(c2c(C)cco2)=O)CC2CC2(CNC(c2sccc2-n2cccc2)=O)C1 78965,c1(NC(=O)Nc2ncc(C(N)=O)s2)nccc(-n2ccnc2)n1 78966,c1(C(=O)NC(C(CO)NC(C(C)Oc2cccnc2)=O)C)sc2ncccc2c1Cl 78967,n1(CC(=O)NCCC(C)NC(C2CC2(Cl)Cl)=O)c(O)nc2ccccc12 78968,CCCCC(F)C(=O)N1CCC(CC(C)NC(=O)C(C)N2CC(C)C2)CC1 78969,C=C(Br)CC(C)(C)C(=O)NC1CN(C(c2cc[nH]c2C2CC2)=O)CCC1C 78970,CC1(CNC(c2cscn2)=O)CCN(C(C2(C)CCCNC2)=O)C1 78971,c1(CC)cc(CC(=O)NCCC(=O)N(CC(C)OC)C(C)C)on1 78972,C1(C(=O)NCC2CN(C(=O)C(C(C)C)N(C)C)CCO2)(OCC)CCSCC1 78973,C(=O)(CC(C)CC(F)(F)F)NC1CCC(C)N(C(C2(O)CCCC(C)(C)C2)=O)C1 78974,C(CC(C)C(=O)NCCC(O)CNC(C1CN(c2nnnn2C)C1)=O)=CCC 78975,S(=O)(=O)(c1ccccc1)N(C)C(N1CCC(c2ccc(F)c(O)c2)CC1)=O 78976,C1(NC(C=CCC)=O)CC(OC)C12CCN(C(C1CCC=CCCC1)=O)CC2 78977,c1(C(=O)NCC(CNC(C2C(C#N)C2)=O)CO)ccc(OCC2CC2)nc1 78978,C1(NC(Cc2n(C)nnc2)=O)CCCCCC1NC(c1ccc(CO)s1)=O 78979,c1(OCC)ccc(Br)cc1CN1CCC(NC(c2cc(CC)[nH]n2)=O)C(O)C1 78980,N1(C(C2(CNC(C3C(CC(C)(C)C)C3)=O)CC=CC2)=O)CC2(CCCC2)C1 78981,C1(NC(C=CC(C)(C)C)=O)CN(C(=O)CNC(c2ccc(Cl)cc2)=O)CC2(CC2)C1 78982,C12(NC(C(C)CC(N)=O)=O)CCC(CNC(c3cccnc3O)=O)(CC1)OC2 78983,c1(C(=O)NCCCCCNC(C2C(C=C)C2)=O)cc(=NS(C)(=O)=O)cc[nH]1 78984,c1(CNC(c2ccc[nH]2)=O)c[nH]nc1C(=O)NCCC1CCOC1 78985,Cc1ncccc1C(N1CC(NC(=O)COC2CCN(C)CC2)C(C(F)F)C1)=O 78986,c1(C(=O)NC(C2CN(C(c3ccccc3C(F)F)=O)C2)C)nc(=O)n(C)[nH]1 78987,C(CCC(C)C(=O)NC(C)C(C)(C)C(=O)NCc1cc(C)nn1C)OC 78988,c1(OCC)ncc(C(=O)NCC2CCN(C(C3CC(O)CN3C)=O)C2)cc1Cl 78989,N1(C(CCN(CCC)C)=O)CC2CC(NC(=O)C=Cc3ccncn3)CC1C2 78990,C(C(C)(C)C1=CCCC1)NC(CC1N(C(C(COC)N(C)C)=O)C2CCC1C2)=O 78991,N1(C(Cn2ncc(C)c2)=O)CC2CCC(NC(=O)CCS(C)=O)CC1C2 78992,c1(C(=O)NCC(C2(O)CN(C(c3ccsn3)=O)C2)(C)C)ccc2[nH]c(=N)oc2c1 78993,C1(CC)(CC)CC(NC(=O)Cc2nocc2C)CN1C(c1ncn2c1CCC2)=O 78994,c1(OC)cncc(C(=O)NCC2CC2NC(C2CC(n3cnnc3)C2)=O)c1 78995,n1(CC(=O)NCC2N(C(C(CO)N(C)C)=O)CCC2)nnc2ccccc12 78996,CC1CNc2ccc(C(=O)N(C(C)CCNC(=O)C(N)=O)C)cc21 78997,CC(=O)CCCC(C)C(=O)NC1(C(N2CCCC2CCCO)=O)CC(O)C1 78998,c1(CC(=O)NC2C(C)N(C(c3n[nH]c4c3COC4)=O)CC2)cccc(F)c1F 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79052,c1(C(=O)NC2C=CC(CC(=O)NCCCN(C)C)C2)cc(O)cc(F)c1 79053,C1(C=C)(C(=O)NCC(CC=C)NC(c2cc(Cl)ccc2N)=O)CCCCC1 79054,N1(C(C(N(C(Cc2nc(C)sc2)=O)C)C2CC2)=O)CC(CO)C1(C)C 79055,C1(NC(C(COC)C)=O)C=CCN(C(=O)CCc2ccc(O)nc2)C1 79056,N1(C(C2(C)CCCCO2)=O)CCOCC(NC(c2c[nH]nc2-c2cccs2)=O)C1 79057,n1(C(C)C)ncc2c(NCCCCC#N)[nH]c(=NCC(C)=C3CC3)nc12 79058,C#CC1(C(N2CCC(OC3CCC3)C2)=O)CCN(C(=O)CC2CN(C(C)=O)C2)C1 79059,Cc1onc(Br)c1C(N1CCC(C(C)NC(c2cccnc2O)=O)C1)=O 79060,CC(C)C(F)(F)CC(=O)NCCN(C(=O)CC1CCC(C)C1)CCOCCO 79061,c1(C(N2C(CNC(c3c(CC)con3)=O)C=CC2)=O)ccc(C(F)F)c(F)c1 79062,C(CC(O)CC(=O)NC1CC(NC(=O)CC(C)O)C1)SC 79063,c1(N2CCC(CC=C)(NC(C3CC4CCCC34)=O)C2)ncnc(Cl)c1C#N 79064,C1(NC(C2C3CN(C(c4cn(CC)nc4C)=O)CC32)=O)CC2(CCC2)C1OC 79065,CC(C)C(CCN(C(=O)CCC1CCCCO1)C)NC(C1(C)CCCO1)=O 79066,CCCN=C(NCc1cc(C)cc(Cl)n1)N1CCN(c2ccccc2F)C(=O)C1 79067,CC(C)(C(=O)NCC(C)(C)NC(=O)CC(F)F)C1CCCCC1 79068,c1(C(=O)NCCC(C)NC(CC(C=C)C)=O)ccc(NCCO)c([N+](=O)[O-])c1 79069,c1(OC)cccc(C(N2CCC2(C)C(=O)NCC2CCN(C)CC2)=O)c1O 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79140,C(CC(C)(C)C)(C(=O)N(C1CC(C#N)C1)CC(=O)N(C1COCC1O)C)OC 79141,c1(NCCOCCNC(=O)CCC(F)F)ncnc2sc(C(F)(F)F)nc12 79142,N1(C(c2c(CC)ocn2)=O)CC2CCC(CNC(C3CC4CCC3C4)=O)C2C1 79143,c1(N2CCC(CCOC)(NC(C3CCC(C)C3)=O)C2)nccc(S(C)(=O)=O)n1 79144,n1(CCC(=O)NCCN(C(=O)C(C)O)CCOC)c(C)csc1=O 79145,CON=Cc1ccc(-c2ccc(OC(F)(F)F)cc2)cc1 79146,N1(c2[nH]c(=NCCC3CC(F)C3)cc(C)n2)CCc2ccc(C#N)cc2C1 79147,N1(C(C(=O)NCC=C)CC2CCOC2)CCCC(c2nn(C)cc2CO)C1 79148,C1(C2(C(N(CCOC(C)=O)C)=O)CC2)CCCN1C(=O)CCn1ccnc1 79149,C(C(CC)CCCC)c1n(-c2c(CC)cccc2)nc(C2CN(C(C)=O)C2)n1 79150,c1(C(=O)NC(C(C)NC(=O)CC(O)CN(C)C)(C)C)ccc(N)c(Cl)n1 79151,C1(CNC(C(CC)CC)=O)CN(C(C2(n3cccn3)CCC2)=O)CC12CCC2 79152,N1(C(C23CN(C(c4ccc(O)nc4)=O)C(C2)CO3)=O)CCN2C(=O)NCC2C1 79153,c1(CCNC(=NCCC)N(C)CCCC(=O)NC)nc2ccc(C)cc2[nH]1 79154,C1(N)CCCCC1OCC(=O)N(CC(CNC(C=CC)=O)(C)C)C 79155,N1(C(CN2C(=O)CNC2=O)=O)C2CCC1CC(NC(C1(F)CCOC1)=O)C2 79156,C(C)(CC(=O)NC12CC(NC(=O)C(C)CC3CC3)(C1)C2)SC 79157,C(=O)(CCCCCCN=[N+]=[N-])N(C1CCN(C(C2CC2(C)C(F)F)=O)C1)CC 79158,CC1CN(C(c2c[nH]nc2-c2cccc(F)c2)=O)CCN1C(=O)C(C)(C)C#N 79159,Cc1nc(O)c(C(N2CC(O)(C(C)NC(=O)CCC(C)(C)F)C2)=O)cc1Br 79160,C(=O)(C(O)C(F)(F)F)NCC(C)N(C(=O)CCNC(c1ccccc1Cl)=O)C 79161,C(CCC)(C(=O)NCc1ncc(C)s1)NC(C(C=C)C)=O 79162,N1(C(C(C2CCOCC2)C)=O)CC=C(C(=O)Nc2c(O)cccc2Cl)CC1 79163,CC(C)(C)C(CNC(c1cccc2nccn12)=O)C(=O)N1CC=CCC1 79164,N1(S(CCCOCC)(=O)=O)CC(C(=O)OC)CCC1C 79165,c1(N2C(C)CC(NC(=O)CCc3ccncn3)C2)ncnc2cc(F)c(F)cc12 79166,C1(C)(C(N2CC(COC)(CNC(C3(F)CCOC3)=O)C2)=O)CC2CC2C1 79167,N1(CC)CCCC(C(N2CCCC2C(C)(C)CNC(=O)CC(C)(F)F)=O)C1 79168,CCC(CN=c1nc2c(cnn2C)c(N(C)Cc2cccc(OC)c2Cl)[nH]1)OC 79169,C(=O)(CC(C(N)=O)NC(C)=O)NCCCC(C)NC(C1(CCOC)CCC1)=O 79170,c1(C(=O)NCC(O)CNC(C2COCCC2(F)F)=O)ccc2ccnn2c1 79171,N1(C(C2(NC(C(COC)C)=O)CCN(C)C2)=O)CCC2(COC(=O)N2)C1 79172,N1(C(c2c(C)cc(F)cc2)=O)CC(C2CN(C(C3(O)COC3)=O)C2)C1 79173,Cc1cc(C(=O)NC23CCOC(CNC(C4CCCCC4C)=O)(C2)C3)ccc1Cl 79174,c1(C(C(N2CCN(C(c3c(C)nsc3)=O)C(C)C2)=O)(C)C)ccccc1[N+](=O)[O-] 79175,c1(SC)ccc(NC(C2CCCN2C(C2CCCN2C2CC2)=O)=O)cn1 79176,CC(C)C(CNC(C1CCN1C)=O)C(=O)N1CCC1c1ccccc1 79177,O=S(=O)(c1cccc(O)n1)N1CCN(c2ccc(F)nc2)CC1 79178,Cc1ocnc1CC(N1CC(C(C)NC(=O)C=CC2CCCO2)C1)=O 79179,C1(NC(CCCCOC)=O)CC2CCC1N(C(=O)CNC(c1nc(C)no1)=O)C2 79180,CCC(CC)C(=O)NC(Cc1cnc[nH]1)C(=O)NCCCNC(=O)C(C)C 79181,c1(C(=O)NC2C(C)CCN(C(=O)C=CBr)C2)nccc2ncccc12 79182,N1(C(CC)=O)CCC(NC(=O)CCCc2cc(C)no2)C(O)C1 79183,C(=O)(C1SCCc2sccc21)NC(CCNC(c1ccnc2c1CCO2)=O)CO 79184,c1(OC(C(=O)NC2(C)CCN(C(c3c(CC)nns3)=O)C2)F)ccc(Cl)c(F)c1 79185,C(C)(CCCNC(=O)Cn1cc(C(F)F)cn1)NC(C1C(COC)C1)=O 79186,c1(C(=O)NC(CC=C)CNC(=O)C(C)CCC)ccc2c(c1)n(C)c(=O)n2C 79187,Cc1occc1S(C)(=O)=NC(=O)C1(C)CNC(=O)N1 79188,c1(C(CNC(C2CCC(CC)C2)=O)O)c(F)cccc1Cl 79189,C(=O)(CC1=CCCCC1)N1CC2(CN(C(C(CC)OC3CCCC3)=O)C2)C1 79190,N1(C(C(C)SCCCC)=O)CCOCC(NC(=O)COc2cccc(Cl)c2)C1 79191,c1(CCC)cc(C(=O)NC2CC(CNC(C3CC34CCC4)=O)CC2O)nn1C 79192,c1(C(=O)NCC2(CN(C(C(CC)SC)=O)C)CC2)cnn(CCO)c1C 79193,Cc1ncc([N+](=O)[O-])n1CC(=O)NCCCCC(CO)NC(c1n[nH]cc1Cl)=O 79194,c1(NC(C)(CCBr)c2nnnn2CC2CCOCC2)cccc2c1CNC2=O 79195,Cc1ccc(S(=O)(=O)NC2CCCNC23CC3)cc1[N+](=O)[O-] 79196,N1(C(C2CC(C)(F)C2)=O)CCN(C(=O)C=CCO)CC2CCCCC12 79197,C1(NC(c2cc(C)c(O)nn2)=O)CCN(C(=O)CN2CCOCC2)CCC1(F)F 79198,C1(NC(C(C2CN(C(=O)CN(CC(C)(C)C)C)C2)OC)=O)CCC2CCC1C2 79199,N1(C(c2c(NC)cncc2)=O)CC2CC(NC(=O)C=CCOC)CC1C2 79200,CC(C)CCCC(=O)N1CC2(CNC(=O)C(O)Cn3cncn3)CC1CO2 79201,N1(C(C2C(CC(C)(C)C)C2)=O)CC=CCC1C(=O)NCC1=CCCC1 79202,c1(C(N2CC(CCC)C(NC(=O)C(c3ccccc3)F)C2)=O)cc(C)cc(O)c1 79203,N1(C(C2C(=C)C2)=O)CCC2(COC(CNC(c3sc4cncn4c3C)=O)C2)C1 79204,c1(NCc2cc(COC)no2)ccc(S(=O)(=O)NC2CCSC(C)C2)c(Br)c1 79205,C1(C(=O)NC2CCN(C(CSCCC(C)C)=O)C2C)CCC2CC1CO2 79206,N1(C(CCCC)=O)CCN(C(C2C(C)C2C)=O)CC1c1cc(F)cc(F)c1 79207,C1(C(=O)NCC(C(C)(C)C)(C)O)CC2(CCN(C(C3(C)C(C)(C)C3(C)C)=O)C2)C1 79208,Cc1oc(CNC(C2CCCC(F)C2)=O)nc1C(=O)N(C1CSC1)C 79209,c1(C(=O)NCC2CC(NC(C3C(C)(CC)C3)=O)C2)cnc(C)n1C(F)F 79210,C1(C(=O)NCCCN(C(=O)CCC2CCCN2C)CCO)(COC)CCOC1 79211,C1(C(N2CCC(c3nn[nH]n3)(C(=O)OCC)CC2)=O)CN(C)CC12CCCN2 79212,c1(CCC)cccc(C(=O)N(C)CC2CCN(C(C34CC(C)C3C4)=O)C2)c1 79213,N1(C(CCC(=O)NC)=O)CCn2nc(CNC(=O)CCC3CCOC3)cc2C1 79214,c1(C(=O)NCCNC(C(C=C=C)C)=O)cc(Br)ccc1N1CCCC1 79215,c1(-c2scc(CC(=O)N(c3ccc(Cl)cn3)C)n2)ccccc1Cl 79216,N1(C(Cn2c(C)ncc2)=O)CCCCCCC1C(=O)NCC1CCCCO1 79217,N1(C(C=CC=CCC)=O)CCC(C)(CCNC(C2(C)CC2(Cl)Cl)=O)CC1 79218,c1(C(=O)NCC2C=CC(NC(CC3(C)CC3)=O)C2)cnc(C(F)(F)F)c(Cl)c1 79219,C1(NC(C(C2CCC2)NC(C=C(C)C)=O)=O)CC(F)(F)C1(C)C 79220,C1(C(N(CC(O)CNC(c2cscc2Cl)=O)C)=O)Cc2nccnc2C1 79221,C1(C(C(=O)N(CCC(=O)N(C2CC2)CC)C)F)CCCCC1 79222,c1(C(N2CCC(OCCNC(CCOC(C)C)=O)C2)=O)ccc(C(F)F)cc1Cl 79223,N1(C(c2[nH]cc(C)c2)=O)CCN(C(c2ccnc(C(C)C)n2)=O)C2CCCCC12 79224,C(=O)(CC(C(F)(F)F)NC(c1[nH]ccc1C)=O)NC(CC)C(=O)NC 79225,C12(CC(N3C(CCNC(CCC)=O)CCC3)=O)COC(C)(C1)C2 79226,C(C1=CCN(C(=O)Cc2ccc(O)cn2)CC1)NC(c1c(SC)n(C)nc1)=O 79227,CC1CCCN(C(=O)CCCCCF)C1CNC(c1cc[nH]c1)=O 79228,n1(CC(CC)O)cc(C(=O)NCC#CCNC(=O)C(C2CCCC2)OC)nn1 79229,c1(C(=O)NCCCCNC(C2C3CCC2(c2cncs2)C3)=O)cccc(Cl)c1F 79230,CC(C)CCCCCC(=O)NCC(C)CNC(=O)C=CC1CCOC1 79231,CCC(C)(C)C(O)C(=O)NCC1(O)CCCN(C(=O)CN2CCCNC2=O)CC1 79232,C1(NC(=O)Cn2cc(CO)nn2)CCC2(CC2)N1C(c1cc(F)ccc1F)=O 79233,C=CCCC(CC(C)C)C(=O)N(CCCCCNC(C1CC12CC(C)(C)C2)=O)C 79234,N1(C(=O)CCCCCl)CCC2(CCCC2N2CCCC(O)C2)CC1 79235,CC1CCN(C(=O)COC2CC=CC2)CC1N(C)C(C1CCOCC1(C)C)=O 79236,C1(CC)(NC(c2ccc(C#N)s2)=O)CCN(C(=O)CCC2CCC(C)O2)CC1 79237,C(c1ccccn1)=C(C)C(=O)NC(C1CCCC1)CNC(C1(C#N)CC=CC1)=O 79238,C(CO)(CCCCNC(=O)C(F)CC1CCCC1)NC(C(c1ccccc1)C)=O 79239,C(c1cccnc1)=CC(N1CCC=CC1C(N1CCC(n2cnnn2)C1)=O)=O 79240,CC1COC(CO)CN1C(=O)CCN(C(=O)CCc1cccs1)CCO 79241,C1(C)(NC(CCN2C(C)CCCC2)=O)CCCN(C(C2CC3CC3C2)=O)C1 79242,Cc1ccc(NC(=O)CN(CCCCNC(=O)C=CC(C)C)CCO)cc1O 79243,c1(CCC)coc(=NCC2(S(=O)(=O)N(C)C)CC2)[nH]1 79244,C1(NC(c2cn(CC)nn2)=O)CN(C(c2ccn(CC)c2C)=O)C(C)(COC)C1 79245,c1(C(N(CC(C)C(=O)NC2CCN(CCF)C2)C)=O)cnn(C)c1Cl 79246,c1(C(=O)NC2(C(F)F)CC2)cnn(-c2ccccc2)c1I 79247,n1(CC(=O)NC(C2CCCN(C(c3cncnc3)=O)C2)C)cc(Br)c(=N)[nH]1 79248,c1(CC(N2CC(C(Cn3cc(CN(C)C4CC4)nn3)F)C2)=O)ccc(O)cc1 79249,c1(NC(C(=O)NCC(C)O)=O)ccc(-c2ncn(C(C)C)n2)cc1 79250,Cc1nc[nH]c1C(=O)NC1(C(=O)NC2CC2CN(C)C(C)C)CC1 79251,c1(CC(N2CC(NC(C(C(CC)O)C)=O)C2)=O)ccc2cccnc2c1 79252,c1(C(=O)NCC2(CCNC(C(C)OCCCC)=O)CC2)nnn2c1CCCC2 79253,C(=O)(C1=COCCC1)NCC1CC(NC(CC2(CS(C)(=O)=O)CC2)=O)C1 79254,C1(C(=O)NC(CNC(C=Cc2cncc(C)c2)=O)CO)CC2(C1)CC(C)(C)C2 79255,N1(C(Cn2ccc(C)n2)=O)CC2(CCC2)CC1CNC(C1COCCN1C)=O 79256,C(=O)(CCCCCC#N)NCC(C)NC(c1cccc(CCCN)c1)=O 79257,N1(C(CCC(CC)NC(=O)Cc2cc[nH]c2)=O)CC2CC3CC2C1C3 79258,N1(C(CC=C=C)=O)CCC2CN(C(=O)CCSc3ccc(Cl)cc3)CCC2C1 79259,c1(C(=O)NC(CCOC)C(=O)NCCCC(C)(C)OC)ccc(Cl)c(F)c1 79260,C(CC(=O)NC(c1ccc(C)nc1)C)(C(F)(F)F)NC(C=CC(CC)C)=O 79261,CC(C)(CNC(=O)C(F)CC1CN(C(=O)CC(C2CC2)C2CC2)C1)C(F)(F)F 79262,CC(CCC(=O)NCC=CC(=O)NC1(CCCc2ncc[nH]2)CCC1)N(C)C 79263,C(N=c1[nH]c(=NCc2ccc(Cl)cc2C)[nH]c2c1CCC2)c1ncc(C)cn1 79264,N1(C(C)CNC(c2cccc(Cl)c2-n2cccn2)=O)C(=O)c2ccccc2C1=O 79265,C1(N(C(CCOCC#C)=O)C)CCCCN(C(=O)CCC2CCCCO2)C1 79266,N1(CCN(C(N(C(c2ccco2)C)C)=O)CCN)CC2CCCCC2C1 79267,C12(NC(Cc3ccn(C)n3)=O)CCCC1N(C(c1cc(F)cnc1O)=O)CC2 79268,C1(NC(CCOCCOC)=O)(CF)CCN(C(=O)CN2CCOC2=O)C1 79269,N1(C(c2c(OC)csc2)=O)CC2=C(C1)CN(C(C1(C(F)(F)F)CC3CC3C1)=O)C2 79270,CCCC(C)CC(=O)NCc1cc(C2CCN(C(c3ccno3)=O)CC2)no1 79271,c1(C(N2CCN(C(C3CCS3(=O)=O)=O)C3C2C3)=O)cc2nc(=O)ccn2[nH]1 79272,N1(C(C2CN(CC)C(=O)C2)=O)C2CCCC1CC(NC(c1csnc1C)=O)C2 79273,Cn1c(C(=O)NC2CCCC(CNC(C3CC4(CC4)C3)=O)C2)cnc1S 79274,c1(C(C)=O)ccc(C(N2CC(NC(=O)C(C)NS(C)(=O)=O)CC2C)=O)cc1C 79275,C(C(F)(F)C(=O)NCC1(C)CCCC1NC(=O)CC1COCCN1C)N(C)C 79276,C1(NC(c2cc(COC)on2)=O)CN(C(C2CCOC2C)=O)CCC12CCC2 79277,c1(C(=O)NCC(C)N(C(=O)C(C)Cc2cnn(C)c2)C)cn2c(n1)COCC2 79278,c1(C(=O)NCC2(NC(C(CC)SC)=O)CCC2)cc(N(C)C)nc(Cl)c1 79279,C=C(Cl)CC(C(=O)NC(c1ncccc1F)C)NC(c1nc(Cl)cs1)=O 79280,c1(C(N2CCC(CCNC(c3c(CCC)nco3)=O)C2)=O)c(C)nnn1CC 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79386,C(N=c1[nH]c(=NCCOC2CCCC2)[nH]c2c1CCCC2)c1c(F)ccc(F)c1 79387,C=CCC(C(=O)NC(CCC)C(O)C(=O)N(C(CC)CC)CCO)C(C)C 79388,c1(CC(=O)N(C(C)C)CCN(C)C(c2c[nH]c(=N)o2)=O)cccnc1Cl 79389,C(N=c1ccnc(NC2COC3(CCCC3)C2)[nH]1)C1C(C)(C)CCO1 79390,C1(NC(C(CC)C(C)C)=O)CCOC2(CCC2)C1 79391,N1(C(c2c(C)cco2)=O)CCCC(C(C)NC(=O)C2=CCCC2)C1 79392,c1(C(=O)NC2CN(C(COCC)=O)C(C)C2)ccc([N+](=O)[O-])cc1 79393,N1(C(COCc2cc(C)no2)=O)C(CNC(C2CCC(=O)N2)=O)CC2COCC12 79394,C1(C(=O)NCC2(F)CC(CO)C2)CCN(C(=O)c2cc(O)ncn2)O1 79395,C1(C2CN(C(=O)CCCCNC(N)=O)C2)(NC(c2cc(C(C)C)no2)=O)CC1 79396,C1(C(=O)NC(C2CCN(C(c3ccncc3N)=O)CC2)C)Cc2ccncc2C1 79397,N1(C(CC2ON=C(C)C2)=O)CC(NC(c2c(N)cccc2Cl)=O)CC(F)C1 79398,CC1CN2CCC1NCc1cc(no1)C2=O.c1(C(N(C)C)=O)csc(C2CC2)n1 79399,CCN=c1cc(C(N2CC3OCC(NC(=O)CN(C)C4CC4)C3C2)=O)cc[nH]1 79400,c1(NC(=O)CCNc2ncc(Cl)cn2)ccc2c(c1)OC(F)(F)O2 79401,C1(CCN)(NCC(C2CC3CCC2C3)C(=O)O)CCOCC1 79402,CC(CC1CCC1)C(=O)NC(C1CN(C(=O)CCc2cc[nH]n2)C1)C 79403,Cc1cnccc1CN(C)C(C1(C(C)NC(=O)CC(C)n2cccn2)CC1)=O 79404,CC(CC(C)(F)F)C(=O)N(CCCCCNC(c1cc2n(n1)CC(F)C2)=O)C 79405,C1(CC(C)NC(=O)C(Cc2ccoc2)NC(=O)CCN(C)C)CCCCC1 79406,S(=O)(=O)(c1ccc(N(C)CCc2ccc(Cl)cc2)c(Cl)c1)NCC(C(C)O)C 79407,C=C(C)CCC(=O)N1CCC(C(C)(C)NC(c2c[nH]cc2-c2ccc(C)s2)=O)C1 79408,c1(C(CC)C)cc(CSC)c[nH]1.C1(=O)CN1S(C)(=O)=O 79409,c1(N2CCC(OCCOCC)C2)nncc2c(C)nn(C)c12 79410,N1(Cc2cnc(C)nc2)CCC2(CC1)CC2C(N1CCC2(CCC2O)C1)=O 79411,c1(OC)cc(SC)ccc1C(=O)NC1C2CC1CN(C(=O)C(C)(O)C1CC1)C2 79412,Cc1cc(OCCCC(=O)NCCNc2ccccn2)ccc1Cl 79413,N1(C(C(C)=CC)=O)CCCCC2(C1)CN(C(=O)CCn1ccnc1C(C)C)C2 79414,c1(C(=O)OC)cc(NC(=O)C(C2CCOC2)NC(=O)OC(C)(C)C)c(C)o1 79415,Cc1cc(C(=O)NC2CC=CCC2C(=O)NC(C)C(=O)NC2CC2)c(N)s1 79416,N1(C(c2c(NC)nccc2)=O)CCCC(NC(c2ccc(N(C)C)cn2)=O)CC1 79417,N1(C(C2C(=O)OCC2)=O)CCC2(CCCCN(C(c3ccc(O)nc3)=O)C2)C1 79418,c1(OC)ccc(C(N2CCN(C(C3CCCSC3)=O)C(C)C2)=O)cc1C 79419,C1(CNC(C2(C#N)CC2)=O)CCCCN1C(C1(C(F)(F)F)CCCCC1)=O 79420,C1(C(=O)NC2(CCCNC(CCCCN(C)C)=O)CC2)CCC2CC2CC1 79421,c1(N2CCC(c3occc3)CC2)nc2cc[nH]c2c(=NCC2CCCO2)[nH]1 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79457,C12(NC(=O)CSC3CC3)CN(C(c3cc[nH]c3)=O)CC1CS(=O)(=O)C2 79458,C(=O)(CC(C)c1ccccc1)NC(C)CNC(=O)C=CCOCC(F)(F)F 79459,c1(C(N2CC(C)C(NC(c3cc4oc(Cl)cc4[nH]3)=O)C2)=O)cn2ccccc2n1 79460,C(=O)(CCC(=O)C(C)(C)C)N1CC(C(=O)NCCc2ncn(C)n2)CC(C)(C)C1 79461,C(=O)(C(CCC1CCC1)NC(=O)CCC=C(C)C)NC(CC)C1CC1 79462,c1(CCC(=O)NCC(CC(C)O)C)ccnc2ccccc12 79463,N1(C(c2cc(C)n(C)c2)=O)CC(NC(c2conc2C(C)(C)C)=O)CCC1C 79464,C1(CC)CN(C(C2CCOCC2(C)C)=O)CCN1C(=O)C=CSc1ccccc1 79465,C(=O)(C1=CCCCO1)NC1CCCC(C(=O)Nc2cc(C)sc2C)C1 79466,C=CC1CN(C(=O)C(C)C2CCCC2)CC1NC(c1cn(C2CCC2)nn1)=O 79467,c1(C(=O)NCC2C(Cn3cc(CC(C)O)nn3)C2(F)F)[nH]c(=N)ccc1Br 79468,C1(C(=O)NC2CC(CNC(c3ccccc3C(N)=O)=O)C2)(OC)CCCC(C)C1 79469,N1(C(c2n(CCCC)ncc2)=O)CC2CC(NC(c3cnoc3C)=O)CC1C2 79470,C1(NC(c2c(CC)cc[nH]2)=O)C2CC3CN(C(c4cnc5sccc5c4)=O)C1C3C2 79471,N1(C(CC2CC(CC)OCC2)=O)CCCN(C(c2cnsn2)=O)CCC1 79472,C(C1c2ccsc2CCN1C(=O)C(O)CC1CCCCC1)NC(CCC=C=C)=O 79473,c1(OC)ccc(S(=O)(=O)N(C)C)cc1NC(c1csc(CO)n1)C(=O)O 79474,Cc1cc(C(=O)NC2COCCN(c3nnc(C4CC4)s3)C2)nc(Cl)c1 79475,C1(CN(C(CSCC(C)C)=O)C)CN(C(=O)CC2COCCN2C)CCO1 79476,N1(C(c2cc(C)ns2)=O)CCC(CNC(=O)CCC2(C)CC2(F)F)C(F)(F)C1 79477,CC1(CNC(c2n[nH]c(C3CC3)n2)=O)CCCN1C(=O)CCC1CCC(=O)N1 79478,Cn1nnc2cc(C(=O)NC3(C)CC(NC(c4c[nH]c(=N)s4)=O)C3)ccc12 79479,C1(CNC(Cc2ccc(C)cc2)=O)CCN(C(=O)CC2(CO)CC2)CC1C(C)C 79480,C(=O)(CC1CCc2ccccc21)NCCN(CCC)C(C12CCC1C2)=O 79481,C1(C(=O)NCC2(C)CCN(C(c3n(C)nc(C4CC4)c3)=O)C2)CN2CCN1CC2 79482,C(C(=O)NCCNC(=O)Cc1ccnc(Br)c1)(C(C)(C)C)N(C)C 79483,c1(C(N2C(C(C)NC(=O)C(C)(Cl)Cl)CCC2)=O)ccc2ccoc2c1 79484,CCC(CCC(=O)NC1CC(NC(=O)CC2OCCC2(C)C)C1)OC 79485,c1(C(C)C)n[nH]cc1C(=O)NC(Cn1ccnn1)C(=O)NC(c1ncn(C)n1)C 79486,c1(N2CCC(C=C)CC2)nc2ccc(S(=O)(=O)NC3CCCC(SC)C3)cc2s1 79487,C1(C(N2C(CN(C(C3CN(C(C)=O)C3)=O)C)CCC2)=O)CCc2nncn2C1 79488,N1(C(C(C(C)NC(=O)Cn2cnnc2)C)=O)C2CCCC1CC2 79489,c1(C(N2CCN(C(c3c(C)nn[nH]3)=O)CC23CC3)=O)cc2c(O)ccc(F)c2[nH]1 79490,c1(OC)c(I)ccc(C(N2CC(c3ccccc3)C(C#N)C2)=O)c1C 79491,c1(CC)n[nH]c(=NC2CCN(C(=O)CCc3cn[nH]c3)CC2)o1 79492,C1(C(=O)NCC2(F)CCN(C(C(F)=C(C)C)=O)CC2)CC(C)(C)OC(C)(C)C1 79493,C1(C(N2CCC(N(C(=O)Cn3nnc(C4CC4)n3)C)CC2)=O)OC2CCC1CC2 79494,c1(C(=O)OC)ccn(CC(=O)NCCN(CC(C)O)C(c2cnccn2)=O)n1 79495,N(C(=NCc1ccc(OC)cc1)NCC12CC(CCO1)C2)C(C#C)C1CCC1 79496,c1(C(=O)NC(CCOC)CNC(=O)CC2(NC(C)=O)CC2)ccnc(C)c1N 79497,c1(C(N2C(C(=O)OCC)CCCC2)C(=O)NCCSC)cc2c(cn1)OCCO2 79498,C=CCCCC(C(=O)NC(CF)C(F)(F)F)NC(=O)C(C)c1cc[nH]n1 79499,N1(C(C2N(CC)CCOC2)=O)CC(C)(C)CC1CNC(=O)CCP(C)(C)=O 79500,Cc1cc(C(=O)N(CCC(=O)NCC2CCC(C)(C)O2)CC2CC2)cn1C 79501,C1(C(=O)Nc2cc(O)n[nH]2)CCCC12CCN(Cc1csc(Br)n1)C2 79502,Cc1cc(=NC(CCO)C2CCSCC2)[nH]c(=NCc2cccc(CO)c2)[nH]1 79503,C1(NC(CNC(CC)=O)=O)(CF)CCN(C(=O)C=C2CCC2)C1 79504,c1(C(=O)NCC2C(NC(c3c(CC)ccs3)=O)COC2)ccc(F)c(C)c1F 79505,C=CC(C)(CC)C(=O)NC(CC(=O)Nc1cnc(N(C)C)nc1)C1CC1 79506,N1(C(c2cn(CC)nc2)=O)CCC2(C)CN(C(=O)CC3CNC(=O)O3)CC12 79507,C1(N(C(C(C2CCCC2)OCC)=O)C)CCCCC1NC(c1ccc(C)nn1)=O 79508,Cc1c(-c2cnc(F)c(C(=O)Nc3cnccc3C(N)=O)c2)cccc1[N+](=O)[O-] 79509,c1(C(=O)NCCCNC(C(CC2CCCCC2)OC)=O)c([N+](=O)[O-])c(C)nn1C 79510,n1(CC)nc(C(C(=O)NCCC2(C)CC2)N(CCS(C)(=O)=O)C)c(C)n1 79511,c1(C(=O)NC2C(C)CN(C(c3ccc(C(N)=O)s3)=O)C2)cccc(S(N)(=O)=O)c1 79512,c1(CC(=O)NCC(n2cc(C3(CO)CCN(C)CC3)nn2)C)c(F)cncc1Cl 79513,c1(C(=O)NC2C(CC)N(C(c3ncc(F)cn3)=O)CC2)cc(=O)cc(Cl)[nH]1 79514,C=C(C)CCCC(=O)NCCCC1CCCN1C(=O)C(N1CCOCC1)C 79515,N1(C(C=CC=CC)=O)CC(CO)C2(C1)CN(C(=O)C(O)Cc1ccccn1)C2 79516,N1(C(CCCCN(C(CCNC(=O)OCC)=O)C)=O)CC2CCCCC2C1C 79517,c1(C(=O)NC2CCC(CCNC(C3(CC(C)C)CC3)=O)C2)cnn2ccsc12 79518,Cc1cc(C(N2CCC(CNC(=O)CN3CCCC3=O)C(C)C2)=O)c(N)c(Cl)c1 79519,c1(OC)cccc(N(C(=O)COC(C)(C)CNC(c2nc(C)oc2C)=O)C)c1 79520,C(CC(O)C(=O)N(CCCCNC(=O)CCC(C)OC)C)SC 79521,Cc1c(CC(=O)N(CC(=O)NOC2CCOC2)C2CC(C#N)C2)cco1 79522,C(=O)(CS(=O)C(F)(F)F)NCC(CCCC)NC(c1cnc2ccoc2c1)=O 79523,c1(C(C)CC(=O)NCC(O)CN(C)C(c2ncn(C)n2)=O)ccc(Br)cc1 79524,N1(C(c2cccc(N(C)C)c2)=O)CCN(C(C2CC(C)(F)C2)=O)C2COCC12 79525,N1(C(=O)OC)CCN(C(C)C(=O)NC2CC(CC#N)C2)C(=O)C1 79526,C12(CCNC(CNC(=O)OCC=C)=O)CCC1CN(C(=O)CC1CC(F)(F)C1)C2 79527,c1(NC(C2(O)CCN(Cc3ncccc3C(F)(F)F)C2)=O)ccccc1I 79528,N1(C(c2cnc(N3CCC(CC4CC4)CC3)cn2)=O)CCC(C2CCOC2)CC1 79529,N1(C(c2n[nH]c(C)c2O)=O)C2CCC1C(C)C(NC(c1ccc(CF)cc1)=O)C2 79530,c1(CC(=O)NC(CC)CNC(=O)C(C)n2cnnn2)ccc(C)c(C)c1 79531,N1(C(=O)CC2(COC(F)(F)F)CC2)CCCC1C1(O)CC1 79532,c1(CNC(C2(NC(C3SCCS3)=O)C(C)C2)=O)ccc(Cl)cc1 79533,C1(C(=O)NCCC(=C)CNC(=O)CC2=CCOCC2)C2CC3CC(C2)CC1C3 79534,C(=O)(C(F)CCC(C)(C)C)NC(C)C(CO)NC(=O)C1=NOC2(CCC2)C1 79535,C(CCCN=C(NC1CCC1)NC1CCCC1)NC(C1(Cl)CCCCC1)=O 79536,c1(CC)nc(C)[nH]c1C(N1CCOC(CN(C(=O)C(C2(O)CCCC2)F)C)C1)=O 79537,C1(C(=O)NCC2C(NC(c3cc(OC)no3)=O)CCC2)CCC(C)(O)CC1 79538,N1(C(CC2(OC)CC2)=O)CC(C(N)=O)OC(C)C1.c1(C(=O)N)cnoc1CS(C)(=O)=O 79539,c1(C(c2ccccc2)NC(=O)CC2CCN(C3CC3)C2)c(F)ccc(O)c1F 79540,Cc1nc(Br)cnc1NC(C1CCCN(C(c2cnnn2C)=O)CC1)=O 79541,C1(OC)CCCC(C(N2CC(F)(CNC(c3c(C)csc3Cl)=O)C2)=O)C1 79542,C[Si]1(C)CCCCN(CC(N2CCC(CCS(N)(=O)=O)CC2)=O)C1 79543,N1(C(c2c(C)nc[nH]2)=O)CCC(F)(F)C(CNC(=O)Cc2ccnc(Br)c2)C1 79544,N1(C(CN(CCCCCC)C)=O)CCOC(C(N(C2(CC)CCC2)C2CC2)=O)C1 79545,C(=O)(CCCCSC)NCC1(OC)CN(C(=O)COC2CCOCC2)C1 79546,C(=O)(C1=CC2CCC1C2)N1CC(F)(CNC(c2cc(OC)no2)=O)C1 79547,C1(CNC(N2CCC(O)C2C2CC2)=O)CC(F)(F)C(=O)N1 79548,C1(NC(CSC)=O)CCCN(C(=O)CC2(O)CCC2)CC1 79549,C1(C(N2CCCC(n3cc(CC(O)C4CC4)nn3)C2)=O)CCCC12CC2 79550,C1(CCC)(NC(=O)CS(=O)(=O)NCC)CCN(C(=O)C2=C(Cl)CC2)CC1 79551,N1(C(C(C)OC)=O)CCCC(C)(NC(C23CC(C(=O)OCC(F)(F)F)(C2)C3)=O)C1 79552,Nc1c(C(N2CCCC(O)(CNC(=O)C=CC3CCCO3)C2)=O)ccc(Cl)c1F 79553,N1(CCC)CCCCC1C(N1CC2CC2(CNC(=O)CSC(F)F)C1)=O 79554,N1(C(CC2C(=O)NC(=N)S2)=O)CC2CC(CNC(=O)Cc3cc(C4CC4)no3)C2C1 79555,c1(COC(C)=O)cccc(-c2cnc(CNC(c3cc(O)ncn3)=O)nc2)c1 79556,C(c1cc(Cl)cc(Cl)c1)=CC(N1CCCCC(CNC(c2cccnc2)=O)C1)=O 79557,C1(C(=O)NC2C3CN(C(CSCC)=O)CC32)CC2(CCC2)CCO1 79558,N1(C(C2(CNC(=O)CC3(OC)CCC3)CC2)=O)CC(OC)C(CC(C)(C)C)C1 79559,C(C)(c1cccs1)=CC(=O)NCCCN(C(C1CC(OC)C1)=O)CCO 79560,N1(C(CC(OCC)OCC)=O)CCN(C(=O)C(=O)N=S(C)(C)=O)C(C)C1C 79561,c1(OC)cc(C(N2CCC3(CC2)CC3NC(=O)C(F)C(C)C)=O)cc2ccoc12 79562,C#CC1(C(=O)N(C)Cc2cc(C)nn2C)CN(C(C2CCOC2)=O)C1 79563,Cc1cnc(N2CCC(NC(=O)CC3CN(C)C3)C2C)nc1 79564,c1(C(N2CCC(c3ccccc3)(COC)C2)C(=O)NCC)cn2ccccc2n1 79565,Cc1cc(Cl)c(C(N2CCC(NC(c3ccc(CO)o3)=O)C(F)C2)=O)cc1C 79566,c1(-c2nc(C(C)C3CC3)nn2C2CCCCC2)cccc2c1CCCC2 79567,c1(OC)cccc(-c2nc(C(c3cccs3)C)n(Cc3cccs3)n2)c1 79568,n1(CC)cnc2c(NCC3(SC)CC3)[nH]c(=NCc3n[nH]c4c3COCC4)nc12 79569,CC1CC(C(=O)NCC(C)NC(=O)Cc2ccco2)CO1 79570,C(=O)(N1CC(O)CCO1)NC(C)CS(C)(=O)=O 79571,N(C(=NC)N1CCC(NC(c2cccs2)=O)C1)CC1N(CC)CCC1 79572,N1(C(C(CC)(C)O)=O)CCC2(CCN(C(c3cc(COC)[nH]n3)=O)CC2)C1 79573,CCCCCCCCN(C)C(C1CCCC1CNC(c1ccc(C(C)=O)o1)=O)=O 79574,Cc1ccc(C(N2CC(NC(=O)CC(C)n3ccc(C)n3)C(O)C2)=O)nc1 79575,C(C)(C(=O)N1CC(NC(=O)C(C)C2(O)CCC2)C1)(c1cccs1)OC 79576,C(=O)(CCCN=[N+]=[N-])NC1(CC=C)CCN(C(C2CCCC(=O)N2C)=O)C1 79577,Cc1ccc(C=CC(N2CCC2CNC(C2CC(=O)N(C(C)(C)C)C2)=O)=O)o1 79578,C1(NC(COC2(C)CCC2)=O)CC2(CCN(C(C3CCC4(CCC4)C3)=O)C2)C1 79579,c1(C(=O)NC(C2CCN(C(C3CCS(=O)(=O)C3)=O)C2)(C)C)csc2nnsc12 79580,C1(NC(=O)CCc2cnc[nH]2)CCCC(NC(c2cscc2F)=O)CC1 79581,C1(C(=O)NCCNC(c2cc(Cn3cc(C)cn3)on2)=O)(COC)CC=CCC1 79582,c1(N(CC(=O)NCCC)C)nc(=NC2CCCCC2)[nH]c2ncn(CC)c12 79583,N1(C(CCSCC)=O)CC2CCN(C(c3cc(COC)no3)=O)CCC2C1 79584,N1(C(C2CCCN2C2CC2)=O)CC2CCCC(C1)N2C(c1cccnc1Cl)=O 79585,NS(=O)(=O)c1cccc(C(=O)NC2CCCC2CNC(=O)CCc2cnc[nH]2)c1 79586,c1(C(=O)NC23CN(C(c4n(C)cnc4)=O)C(C2)C3)ccc2c(c1)CC2 79587,c1(C(=O)NC2CCCN(Cc3c(C)ccnc3)C2)cc2cc(Cl)ccc2[nH]1 79588,c1(C(N(CCC(C)NC(c2c(CC)con2)=O)C)=O)csc2ccc(F)cc12 79589,N1(C(C(C(CC)C)=O)=O)C2CCC(C(=O)NCc3cc(C)[nH]n3)C1CC2 79590,c1(CC)cc(C(N2CCCC2(C)CNC(=O)C=CCOC)=O)c2c(c1)CCO2 79591,CC(C)(CO)C(=O)NC1CCN(C(c2cnc(C(F)(F)F)o2)=O)C1 79592,CC1(C)C(NC(=O)C(O)CC2CCOCC2)CCN1C(C1CCS(=O)(=O)CC1)=O 79593,N1(C(CN2C(C)CCC2)=O)CCCC(O)(CN(C)C(c2cccnc2CO)=O)C1 79594,CC1OC2(CNC(=O)C=Cc3ccccn3)CC1(NC(C1CCCN1C)=O)C2 79595,c1(CC(=O)NCCCN(CCCOCC(=O)OC)C)ccc(C)c(C)c1 79596,N1(C(C2C(OC)CCCC2)=O)CC2CCC1CN2C(=O)CCCC1CCCO1 79597,N1(C(c2c(C)[nH]nc2C(F)F)=O)CCC(NC(=O)OC(C)(C)C)CC(C)(C)C1 79598,C1(C(N2C(CN(C)C)COCC2)=O)CCN(C(=O)C=CC2CC2)C1(C)C 79599,c1(C(=O)NCC(CS(C)(=O)=O)(F)F)cc(Br)cc2c1CCCC2 79600,c1(C(N2CC(O)CC(NC(c3cccc(CO)c3)=O)C2)=O)ccnc2ccsc12 79601,C1(CNC(C(CC2CCC2)NC(=O)CSCC(F)F)=O)CC(O)CCO1 79602,c1(C(=O)NCCN2CCC3CCCC23)cncc2n[nH]cc12 79603,Cc1cc2ccc(C(=O)NCC3CCN(C(=O)CCC4CC4(Cl)Cl)CC3)cn2c1 79604,C1(NC(C(c2ccccn2)C)=O)CCN(C(c2ccc(=O)oc2)=O)CC12CCC2 79605,c1(C(=O)NC(CNC(CC(C)c2ccncc2)=O)(C)C2CCC2)cc(Cl)cn1C 79606,c1(C(N2CCC(NC(C=CC(C)(C)SC)=O)C(F)C2)=O)ccc(N)c(Cl)c1O 79607,N1(C(C2CNC(=O)N2)=O)CCN(C(c2cnn(C3CCCC3)c2)=O)C2COCC12 79608,C1(CNC(C(CC)OCC)=O)CCCC(CNC(=O)C=Cc2nc(C)co2)C1 79609,c1(C(=O)NCC(CNC(c2c(C)ccnc2)=O)C)cccc2occ(Br)c12 79610,C(C(=O)NC(C)(C)C(C)NC(=O)Cc1cscn1)(C(C)C)n1ncc(C)c1 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79800,c1(CNC(C2C(c3ccc(C(=O)OC)cc3)C2)=O)ccc(F)cc1Cl 79801,N1(C(C(CCC)NC(c2ccc(C#C)cc2)=O)=O)CC(C)(C)CCC1C 79802,C1(C(=O)NCC(C2CC2)NC(Cn2cc(C(C)=O)nn2)=O)CCC2(CCC2)O1 79803,C12(C(=O)NCC3N(C(CC4C(CC)C4)=O)CC(F)C3)CCCN(CCC1)C2 79804,C1(N(C(C(C)C)=O)C)CCCCN(C(C2(c3cccnc3Cl)CC2)=O)C1 79805,Cc1ccncc1C(C)NC(c1nc(CNC(c2cc(C)c(C)[nH]2)=O)oc1C)=O 79806,N1(C(=O)NCCOCCCC)CCC(CC#N)C(F)(F)CC1 79807,C(=O)(C1CCCc2sccc21)N1C2C(NC(C3C(CCC)CCC3)=O)C(C2)C1 79808,C(=O)(C1=Cc2ccccc2C1)N(CCOCCNC(CCC(C)OCC)=O)C 79809,c1(C(N2CCN(C(C3N(C)CCCC3)=O)C(C)C2)=O)ccc(Cl)c2[nH]ccc12 79810,Cc1n[nH]cc1C(=O)NC(C)CCN(C(=O)CC1(O)CCOC1)C 79811,C1(C(N(C2CCN(C(C(CN(C)C)(C)C)=O)C2)C)=O)CC2CCC(C1)N2C 79812,c1(CNC(C2C3CN(C(C(C)Cc4ccco4)=O)CC32)=O)cc(F)ccc1[N+](=O)[O-] 79813,c1(C(=O)NCCCNC(C2(Oc3ccc(Cl)cc3)CC2)=O)cccc2c1CCO2 79814,c1(-c2cc(C(=O)Nc3c(SC(C)(C)C)cccc3)no2)ccc(Br)cc1[N+](=O)[O-] 79815,C1(NC(C(C)(C)n2cc(Cl)cn2)=O)CCC(O)CN(C(C2CC2F)=O)C1 79816,C1(S(N)(=O)=O)(C(=O)NCCCCCNC(c2c(SC)cnn2C)=O)CCC1 79817,C(=O)(C(C(=O)N1CCN(C)CC1CNC(=O)CCCCC(C)=O)C(C)(C)C)OCC 79818,Cc1cccc2[nH]cc(CCC(=O)NCC(CC(C)C)NC(c3cc[nH]n3)=O)c12 79819,c1(C(=O)NCC(C)(C2CCC2)NC(COCCC=C)=O)c(C)ncn1O 79820,c1(CC)nc(C(=O)NC2CCC(CC(=O)N(C)Cc3cc(=O)cc[nH]3)C2)c(C)o1 79821,c1(SCC(=O)Nc2cccs2)cc(C(=O)O)co1 79822,N1(C(c2c(CC)nc[nH]2)=O)CCN(C(c2cc(C)on2)=O)C2(CCC2)C1 79823,C1(NC(COCCC#C)=O)CS(=O)(=O)CC1NC(c1cc(OCC)ns1)=O 79824,C(=O)(CCC(C)(C)F)NC(C1OCCN(C(c2nc(C)n(C)n2)=O)C1)C 79825,N1(C(C(C)(C)OCC)=O)CC2(CC(NC(c3ccc(CO)nc3)=O)CO2)C1 79826,c1(C(=O)NC2CCCN(C(CSCC#C)=O)C2C)ccc2c(c1)N(C)C(=O)CO2 79827,C1(CCC)CCCN(C(=O)C(CC(F)F)N(C(=O)C(C)OC(C)(C)C)C)CC1 79828,Cc1cc(CNC2CCC(C(=O)Nc3ccc(Cl)cc3I)C2)cc(O)c1 79829,c1(C(N2CC(NC(C3C=CCCC3)=O)C3(C2)CC3)=O)n[nH]c2ccccc12 79830,CCC(CC(=O)NC1CC=C(C(=O)NCC2CC3(CCC3O)C2)C1)C(F)F 79831,N1(C(C(CC)(C)F)=O)CCC(C2CCN(C(c3cc(C)cc(C)c3N)=O)C2)CC1 79832,N1(CCC)CC(C(=O)NCCCCN(C(=O)CC2CC2(Cl)Cl)C)CC1=O 79833,c1(C(=O)NC2C(NC(C3(C)CC3)=O)COC2)ccnc(OC2CCOC2)c1 79834,N1(C(c2cc(C)c(C)nn2)=O)CC2OCC(NC(C3CC(C)C3)=O)C2C1 79835,C1(C(=O)NCC2C(C)CN(C(=O)C(C)OCCN(C)C)C2)CCCC(C)(C)C1 79836,N(C(=NCCCCl)NCc1ccc2c[nH]nc2c1)CC(COC)(C)C 79837,C1(N(C)C(C2CC(C)(C)C2)=O)CCCCN(C(C2(N(C)C)CCCSC2)=O)C1 79838,n1(C(COCC)(C)C)ccc(=NC(=O)OC(C)(C)C)[nH]1.C1(C)C(CO)N1 79839,c1(COC(C(=O)N(C(C)CN(C)C(c2sccc2F)=O)C)C)ccc(Cl)cc1 79840,N#Cc1ccc(NC(=O)NC(=O)C(c2ccccc2)Sc2ccc(Br)cc2)cc1 79841,C=C(C)C1CN(C(=O)C(=O)NCCN(C(=O)C(C)OCCOC)CC2CC2)CCO1 79842,N1(C(CCCCCC)=O)CCC2(CC1)COC(CNC(=O)C(C)(CC)OC)C2 79843,c1(C(N(CCC[Si](C)(C)C)C)=O)ccn2ncc(Br)c2c1 79844,c1(NC)cnncc1C(N1CCC(NC(=O)C(CO)N(C)C)C1)=O.CN 79845,C1(NC(C2CC(O)(CC#C)C2)=O)CN(C(c2cn(C)nc2C)=O)CC2CCCC12 79846,c1(SC)ccc(C)c(NC(=O)NCC2(O)CCS(=O)(=O)C2)c1 79847,C1(CNC(c2cccc(OC)n2)=O)CCN(C(=O)C(C)(F)F)CC1O 79848,CCCCCCCCCC(O)CC(=O)N1C2CC1CN(C(=O)C(O)C(C)CC)C2 79849,C(C(=O)NCCOC)(C1CC1)NCC1CC1.C(=O)(C(C)OC)OCCO 79850,CC1(CNC(C2CC=CCC2C(F)(F)F)=O)CCN(C(c2csc(=N)[nH]2)=O)CC1 79851,C1(C(N2C(CC(=O)NCc3cnc(CC)s3)CCCC2)=O)C2C3CCC(C3)C12 79852,C=C(C)CCC(C)N=c1[nH]c(=NCC2(C)CC2(Cl)Cl)c2ccc(C)cc2[nH]1 79853,c1(C(=O)NC(C)Cn2cc(CC(O)C3CC3)nn2)cc2oc(Br)cc2s1 79854,c1(-c2ncc(C(N(C(CNC(C(C)OC)=O)C)C)=O)s2)ccccc1Cl 79855,C(=O)(CCCNC(C1CCC1)=O)NCC(C)C.C1(C)(C)CNC(=O)C(C)N1C 79856,Cc1ccnc2c(C(N3CCC4CN(C(=O)C(O)CC(N)=O)CCC34)=O)cnn12 79857,C(=O)(C(C)(C)C1=CCN(C(=O)C(C)CCCC(C)C)C1)NCC(C1CCC1)OC 79858,N1(C(CC(C)C2CCCO2)=O)C2CCC1CC(NC(=O)C(C)(C)c1cscn1)C2 79859,N1(C(c2c[nH]nc2C2CC2)=O)CCN(C(C2(C3CCC3)CC2)=O)C2CCCC12 79860,CC1CCC(CC(N2CCCC(CN(C)C(c3nnn(C)n3)=O)C2)=O)CC1 79861,C1(NC(c2cc(C)cc(Cl)c2)=O)CS(=O)(=O)C2CN(C(C3CSC3)=O)CC12 79862,N1(C(C2CCN(C(c3c(CC)con3)=O)C2C(C)C)=O)CCC(C2CCC2)CC1 79863,c1(CCNC(C(C)(C)C)c2nnnn2Cc2ccccc2)ccc(F)cc1Cl 79864,Cc1cnc(NC(C2CN(C(=O)C(Cl)(Cl)Cl)CCC2O)=O)c(C)c1 79865,C1(C(=O)N(CC(C)(C)NC(c2ccc(C)c(C)n2)=O)C)(CC)CCC(O)CC1 79866,CC1CN(C(C2CCC(C)(C)N(C(=O)C(C)(O)C3CCC3)C2)=O)Cc2c[nH]nc21 79867,N1(C(CC(CC)O)=O)CCN(C(c2ocnc2C(F)F)=O)CCC1C 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79886,c1(CNC(C=CC2N(C(C(CC)CN(C)C)=O)CCC2)=O)ccc(F)cc1F 79887,C1(NC(CNC(=O)OC)=O)CCOC12CCN(C(c1cc(=O)n(C)o1)=O)CC2 79888,Cn1cccc1-c1cn(CCCC(=O)NC(=N)O)nn1.C1C(C(=O)O)SC(=S)S1 79889,Cc1nnc2cc(NCC3CCCC(CNC(C4(COC(C)=O)CC4)=O)C3)ncn12 79890,N1(C(C(CC)O)=O)CCC(n2cc(COc3ncccn3)nn2)CC1 79891,CCC(F)(F)C(C)(C)C(=O)N1CC2CCC1CN(C(c1[nH]cnc1C)=O)C2 79892,N1(C(C2CC(=O)C2)=O)CCC2C1CCCN2C(=O)C=Cc1ccccc1[N+](=O)[O-] 79893,C12(c3n(CCC)ccn3)COCC1CN(c1nc(-c3ccccc3)cs1)C2 79894,c1(C(C(=O)Nc2ccccc2)N(C(C(=O)OCC)CC)C)cc(C)nn1CC 79895,c1(C(=O)NCCCC(=O)NC(CC(=O)OCC)C)cccc(C)c1O 79896,c1(C(N2CCC(C(C)(C)C)(CNC(CC3(OC)CC3)=O)C2)=O)cc(C)nc(C)c1 79897,CON(C)CCCNC(C1C=CCCN1C(=O)CC1(C(=C)F)CCC1)=O 79898,C(CCCCC(=O)NC(C)C(C(C)C)NC(C1CCSCC1)=O)OC 79899,O=C(CC1C(=O)Nc2cc(Cl)ccc21)OC1CCOC(c2cccnc2)C1 79900,C(CC(C)C)(C(=O)N1CCCCC(NC(c2occc2C(C)C)=O)C1)NC(C)=O 79901,c1(C(=O)NCC2(COC)CN(C(C3C(C)(CC)C3)=O)C2)c(C)nc(C)n1O 79902,c1(C(=O)NCC2C(NC(=O)Cn3cncn3)C2)c[nH]cc1C1CC1 79903,C1(C)(CC)CCCN(C(C2(CNC(c3cnc(C4CC4)o3)=O)CC2)=O)CC1 79904,C1(NC(=O)NCC2CCN(C(=O)OCC)C2)CCC=CCCC1 79905,C1(C(N2CC(OCc3ccc(-n4cc(Br)cn4)nn3)C2)=O)C2CCCOC12 79906,C1(OC(C2(CNC(COC(CC)(C)C)=O)CC2)=O)CCCC(CO)C1 79907,C1(CC(=O)NCc2cccc(Cl)c2)CCCN(C(C2CC(F)(F)C2)=O)C1 79908,C=C(C)CCCN=c1c(Br)ccc(I)c2ccccc12 79909,C1(C(N2C(CNC(CCC#C)=O)CN(C)CC2)=O)CCC(S(C)(=O)=O)CC1 79910,C1(NC(C2C(CNC(c3c(CC)oc(C)c3)=O)CCC2)=O)CC2CC1C(O)C2O 79911,C1(CNC(C(CCCC)O)=O)CCC12CCN(C(c1cnc(C)[nH]1)=O)CC2 79912,N1(C(C=CC2N(C)CCC2)=O)CCN(C(c2cc[nH]c(=N)c2)=O)CC1CC(F)F 79913,C1(CC(=O)NCCN(CC)Cc2ncc[nH]2)CC1C1CC1 79914,C1(NC(C(C)C2CC2)=O)CN(C(c2cn(C)nc2Br)=O)CCC12CCC2 79915,CC1CN(C(c2cn(C)c(=O)cn2)=O)CCC1NC(c1ccccc1O)=O 79916,C1(COC)(NC(=O)CC2CN(C(=O)CSc3nc[nH]n3)C2)CCC1 79917,CCC(O)C(C)C(=O)N(CC)CC1C(COC)C1(F)F.C12CCN(CC1)C2=O 79918,C1(NC(c2ccc(F)c(Br)c2)=O)CC2CC1N(C(c1ccc(C3CC3)o1)=O)C2 79919,CC(O)C(C(=O)NCCC1CCCN(C(c2csc(Cl)n2)=O)C1)N(C)C 79920,Cc1ccc2c(=NC3CCOCC3C)[nH]c(=NCC3(n4ccnn4)CC3)[nH]c2c1 79921,c1(CCC)ncc(C(=O)NC2CCC(NC(=O)CSc3nncn3C(C)C)C2)s1 79922,C(=O)(C#CC1CCOC1)N1CCCC(N(C(Cc2nc(C)c(C)s2)=O)CCO)C1 79923,C12(NC(COCCOC)=O)CCCCCC1N(C(C1CCCCC(C)(C)C1)=O)CC2 79924,c1(NC(C(C(C)C)NC(=O)Cc2ccns2)=O)ccc(F)cc1CO 79925,c1(C(=O)NCC(C)N(C(c2ccc(N)c(O)c2)=O)CC)ccc2c(C)[nH]nc2c1 79926,C1(C(N(C)CC2(O)CCN(C(Cn3c(C)csc3=O)=O)C2)=O)C2CCC(F)(F)C12 79927,c1(CNC(=O)NC2CC(C(N)=O)OCC2)cc(O)cc(Br)c1 79928,CC1COc2ccc(C(=O)NC3CCC3NC(=O)CCCc3ccsc3)cc21 79929,c1(OC)cc(C(C)=O)c(C(=O)NCC2(N(C)CC3CCCOC3)CC2)cn1 79930,C1(NC(COCCCC)=O)(CO)CN(C(=O)C(C)C2CCCO2)C1 79931,C1(CC(N2CC(O)(CN(C(=O)C(C)(C)C3CCOC3)C)C2)=O)OC(C)(C)OC1=O 79932,C(=O)(C(C)C(O)CC(C)C)NCC(C)(C)OCC(=O)NCC1CC(OC)C1(C)C 79933,C(=O)(C(CC(C)C)CC(C)C)NC1CC2CN(C(CC(C)SC)=O)C1C2 79934,C1(C(=O)NCC(CNC(CNS(CCCOC)(=O)=O)=O)C)CC2(C1)CC21CCC1 79935,C1(CCNC(c2ccc(CO)o2)=O)(OC)CN(C(c2cn(CCO)nn2)=O)C1 79936,n1(CC)ccc(CN(C)C(C2CC(CNC(=O)C(C)OC(C)=O)C2)=O)n1 79937,C1(CCC)COCCN1C(=O)C(C)C(C)NC(=O)C=C(C)C 79938,C1(NC(c2ncc(F)cn2)=O)CN(C(C2CN3CCC2CC3)=O)CC12CCCC2 79939,C1(CNC(CC(C)C)=O)CN(C(C2CCN(C)CC2)=O)CC(C(F)(F)F)O1 79940,C1(C(=O)NC2CC(CCC(=O)NC(C(=O)NCC)C)C2)COC(=O)N1C 79941,C1(NC(C(CC)C(C)C)=O)CC12CCN(C(=O)Cc1ccnc(OC)c1)CC2 79942,N1(C(C(C)C2CC2)=O)CCCC12CCN(C(C1CCOC1)=O)C2 79943,C1(NC(Cc2ccc(C)nc2)=O)CC2CC(C1)N(C(=O)CCc1cccs1)C2 79944,c1(CNC(=O)NC(CC=C)CC=C)noc2c1CCC2 79945,c1(C(N(C(=O)CCc2cccs2)C2CC2)=O)nccc(-c2cnccn2)n1 79946,N1(C(CCCCCC)=O)CCN(C(=O)CCc2cccc(C#N)c2)C(C)CC1C 79947,Cc1[nH]nc2cc(C(N3CCOCC(NC(=O)C(C)C4=CCCC4)C3)=O)ccc12 79948,C1(C(C)NC(C2(C3CCCO3)CC2)=O)COCCN1C(c1cccc(CO)c1)=O 79949,c1(C(=O)NC(C(CCC)O)CO)cc2[nH]nnc2cc1OC 79950,C1(C(N(CCCF)CC)=O)CC(=O)CN1C(c1cc[nH]c1C)=O 79951,N1(C(CCCCN(C(=O)OC(C)(C)C)CC)=O)CCCC(n2nncc2I)C1 79952,CCCCCCC(O)CCC(=O)NC1(C)CCCN(C(=O)CC2OCCO2)C1 79953,N1(C(C2NC(=O)OC2)=O)CC2CN(C(c3cc4n(n3)CCCN4)=O)CC2C1 79954,C(=O)(C1SCc2cccnc21)N1CCN(C(c2c(C)cn(C(C)C)c2)=O)CC1 79955,C1(N(C(=O)C(C)C2CCCO2)CC)CCN(CCOCc2cccc(C)c2)CC1 79956,CN=c1ccc(C(=O)N(C(C)CNC(c2csc(C3CCCO3)n2)=O)C)c[nH]1 79957,C(=O)(C(C)S(=O)Cc1nncn1C)Nc1c(CCC(C)C)cccc1 79958,N1(C(C(CCO)N(C)C)=O)CC(C2CCN(C(C3CC3(C)C)=O)CC2)C1 79959,N(C(=NCCCOC(C)C)N(C)Cc1cc(C)on1)C(c1cccc(Cl)c1)C#C 79960,CC1(NC(c2cc(-c3ccoc3)[nH]n2)=O)CCCN(C(=O)CC2CCC(=O)N2)C1 79961,CCS(=O)(=O)CC(=O)NCC1C(C(=O)Nc2ccc(O)c(C(N)=O)c2)C1(C)C 79962,Cc1cnc(N2CCC(CNC(=O)C(C)C(C)(C)C)C2)nc1S(C)(=O)=O 79963,c1(C(=O)NC2CN(Cc3ccc(Br)nc3)CC2F)ccnc(Cl)c1Cl 79964,c1(C(=O)NCC(CC=C)NC(=O)Cc2cc(C)cc(C)c2)cc(OC)ccc1C 79965,C(=O)(C1=CCCS1)NC1(CNC(=O)CCC2CCC(C(=O)OC)O2)CCC1 79966,c1(C(N2CC3(C(NC(CS(CC)=O)=O)CC3)C2)=O)c(C)cc(O)nc1C 79967,Cc1cc(F)ccc1C(=O)NC(c1csc(-c2cnn(CC3CC3)c2)n1)C 79968,N1(C(C(C2CCCC2)NC(CC2(C)CC2)=O)=O)CCC(CO)C(C)C1 79969,C1(NC(CN(C)C)=O)CCCC1CNC(C1CSCN1C(=O)OC(C)(C)C)=O 79970,C1(C(N2C(CNC(c3cc(Cl)ccc3F)=O)CC2)=O)Cc2ccccc2N1 79971,c1(C(N2C(C)CC(CC(=O)N(CC(COC)C)C)C2)=O)ccc(C#N)cn1 79972,C12(CNC(=O)C3=COCC3)CCCC(CN1C(c1cc(CO)[nH]n1)=O)C2 79973,C(=O)(C(F)CCC(C)C)N1CCN(C(Cc2c(CC)con2)=O)C(CCOC)C1 79974,C=CC1(C(N2CCC(C)(CC(=O)NCC3CCCOC3)C2)=O)CCCC1 79975,C1(CC(=O)NCc2cc(C)ncn2)CCCN(C(c2cc(C3CC3)on2)=O)CC1 79976,c1(C(N(c2nccn2C)CCNC(C(C(=O)OC)C)=O)=O)ccc2nccn2n1 79977,c1(C(=O)NC2CC(NC(C3COCC(C)(C)O3)=O)C2)c[nH]c2c(C#N)cccc12 79978,C(=O)(C(C(C)C)n1cnnn1)NC1C(NC(CC(OCC)OCC)=O)CC1 79979,N(C1CCCc2c(C)cc(C)cc21)CC(CCC)CO 79980,c1(C(=O)NC2C(C)CN(C(C3CCCO3)=O)C2)cc2cccc(Br)c2[nH]1 79981,C1(C)(CC)C=C(C(=O)NC(C)CC2CN(C(=O)C(O)Cc3ccccc3)C2)C1 79982,C1(OC)CC(COc2ccccn2)N(C(c2cnc(Cl)s2)C(=O)NC2(C)CC2)C1 79983,Cc1ncncc1C(=O)NC1CN(C(c2occc2CN(C)C)=O)CC1F 79984,C(CC1=CCN(C(C2CC23CC(C)(C)C3)=O)CC1)NC(CCCC(=C)C)=O 79985,N1(C(C(CCC)N(C)C)=O)C2CCC1C(C)C(NC(=O)C1=C(C)S(=O)(=O)CC1)C2 79986,c1(SC)ccc2cc(C(=O)NC3COC(C(F)(F)F)CN3C(C)=O)[nH]c2c1 79987,c1(C(=O)NC2CC(N(C(CC)=O)C)C2)ccc(OC)c(F)c1N 79988,CCC(CC)C(C(=O)NC(CC1CCCC1)C(N1CCCOCC1C)=O)OC 79989,Cc1cc(CC(=O)N(CCCCNC(C2CCSC(C)C2)=O)C)c(C)s1 79990,n1(CC(C)C)cc(NC(c2ccn(C)n2)c2nnnn2Cc2cccs2)cn1 79991,c1(NC(C2C(NC(=O)COCCc3cc[nH]n3)CCC2)=O)cccc(F)c1F 79992,c1(N(C)C)ccncc1CNC(C1CCCC1NC(=O)CC(C)(C)N(C)C)=O 79993,C1(C(C)C)CCc2[nH]nc(C(=O)NC3(CNC(=O)C(O)CCN(C)C)CC3)c2C1 79994,CC1(C)CN(C(c2csc(C(F)F)n2)=O)C(CNC(C2(Cl)CC23CCC3)=O)CO1 79995,C(C(CO)(CO)NC(C1CCN1S(C)(=O)=O)=O)N(C(c1nc(CC)sc1)=O)C 79996,C12(NC(COCCSC)=O)CCCC1CN(C(=O)C(=O)NCC1CC1)C2 79997,N1(C(C=CC)=O)CCC(CO)C(NC(=O)Cc2cccc(C(F)(F)F)c2)C1 79998,N1(C(c2c(CC)noc2)=O)CC2CCC2(CNC(=O)C(C)(C)COC)C1 79999,N1(C(=O)C=Cc2ccncn2)CCN(C(C2(O)CC2)=O)CC(O)C1 80000,C(=O)(CC(C)CCCCCCC)N1CCN(C(C(C)=CC)=O)C(CCCC)C1 80001,C1(C(NOCCCCC)=O)CC(C)CN1C(=O)C(=O)NOC 80002,Nc1cc2[nH]cnc2cc1C(N1CCC(NC(=O)Cc2csc3cncn23)C1)=O 80003,C(C(O)CC(=O)NCCC1(C)CCOCC1)NC(C(C)OCC=C)=O 80004,C(=O)(C(C)(C)C(F)(F)F)N1CCCCC(CNC(C(C)OC2CCCC2)=O)C1 80005,C1(C(=O)Nc2c(C#N)cccc2)CN(Cc2cc3ncccc3[nH]2)CCC1(F)F 80006,C(=O)(C1=CS(=O)CCC1)N1CCC(NC(c2cn(C(F)(F)CO)nn2)=O)C1 80007,N1(C(CN2CC(C)(OC)C2)=O)CC(CNC(=O)C=CC2CCCC2)CC1C 80008,C12(NC(CC3(C)CC3)=O)CCCC1N(C(c1cnc(Cl)s1)=O)CCC2 80009,C(=O)(C1CCc2cc(Br)ccc21)NCCn1cc(C2CCCN(C)C2)nn1 80010,Cc1scc(C(N2CC3C(CNC(c4ccoc4C4CC4)=O)C3C2)=O)c1N 80011,c1(C(=O)NC(CCC)CC)ccc(=N)[nH]n1 80012,c1(CNC(c2csc(C)c2C)c2n(CC)nnn2)cccc(F)c1 80013,Cc1cc(C(=O)NCCC(O)CNC(c2nscc2Br)=O)ccc1O 80014,C(C(=O)NN1CCCC1C(N1C(C)CC1(C)C)=O)SC(C)C 80015,C(=O)(C1CCCc2ccccc21)NC(C1N(C(Cc2cnc(C)[nH]2)=O)CCC1)C 80016,c1(C(N2CC(O)(C(C)NC(C3CCCN3C)=O)C2)=O)ccccc1Br 80017,C1(NC(=O)C=C2CCC2)CC2CCC1N(C(C1(O)COC1)=O)C2 80018,c1(C(=O)NN2C(Cn3cc(C(c4noc(C)n4)C)nn3)C=CC2)cc(Br)sc1Cl 80019,Cc1cc(CNC(C2(C)C=CCN2C(=O)C(C)c2ccsc2)=O)ccc1F 80020,N1(C(Cn2c(C)ccn2)=O)Cc2nccn2CC(NC(=O)OC(C)(C)C)C1 80021,c1(OC)cc(Br)c(C(=O)NC2CC2CNC(=O)CC(F)F)cc1F 80022,N1(C(c2ccn3cncc3c2)=O)CCCC2(CCCN2C(=O)C=CI)C1 80023,C1(NC(C2CC=C(C)CC2)=O)CCN(C(c2ccn(CCO)c2C)=O)C(C)C1 80024,c1(C(=O)NCCCC(C)NC(C2(OC)CCOC2)=O)cccc2cc(F)ccc12 80025,N1(C(C(C)=C(CC)C)=O)CC(F)CC1CNC(=O)COc1ccccc1C 80026,CC(C(C)(C)C(=O)NCCOC1CC2(C1)OCCO2)NC(=O)OC(C)(C)C 80027,c1(CNC(=O)CC2(NC(=O)C(O)Cn3cncn3)CC2)ccccc1F 80028,CC1CCN(C(C2CC(=O)N(O)C2)=O)CCN1C(c1cc(-c2ccco2)[nH]n1)=O 80029,c1(SCC(=O)NCCC2CCN(C(C3(O)CCOC3)=O)C2)nc2ccccc2[nH]1 80030,c1(C(=O)NCCN(C(CCc2onc(C(C)OC)n2)=O)C)cnncc1O 80031,C1(C(=O)NCC(CNC(c2ccn(CCN(C)C)n2)=O)O)CC2C=CCC(C1)C2 80032,Cn1nc(Br)c2c(NC3CC(=C4CC4)C3)ncnc12 80033,c1(C(=O)NCC(C(C)C)NC(C2(CC(C)C)CCC2)=O)ncccc1C(C)(C)C 80034,N1(C(=O)NCC(C2CC(F)(F)C2)OC)CCC2(CC1)OCCO2 80035,N1(C(CCc2onc(C)n2)=O)CC2(C1)C(NC(=O)CC(C)C(F)F)CCS2(=O)=O 80036,c1(-c2n(CCOC)ccn2)ccc(OC)c(-c2ccc(=NC)[nH]c2)c1 80037,n1(CC)c(N)c(C(=O)COC(=O)Cc2ccc3c(c2)CCC3)c(O)nc1=O 80038,c1(C(=O)NCc2cc(C)c(C(N3CC(F)C(F)C3)=O)o2)cc2ccncc2[nH]1 80039,O=C(C1=CC2CCC(C1)C2)N1CCC2(CC1)CN(C(c1cnc(O)s1)=O)C2 80040,c1(OCC(=O)NCC2N(C(CC(C=C)CC)=O)CCC2)cccc([N+](=O)[O-])c1 80041,CC(O)C(C(N)=O)NC(=O)COC1CCN(C(=O)CC2(O)CCCC2)C1 80042,C1(C(=O)NC2(C)CN(C(c3cc(SC(C)(C)C)ncc3)=O)C2)CC2C(C1)C2(F)F 80043,C1(C(N2CC(SC)C(NC(=O)COCCN(C)C)C2)=O)CC2C(C1)C2(C)C 80044,O=S(=O)(c1ccc(N2CCC(C3CC3)C2)c(Br)c1)NC(c1cccnc1)C1CC1 80045,c1(SCC(=O)NC(CCN(C(C(CC)F)=O)C)C)ccc(F)c(F)c1 80046,Cc1cc(C(N2CC(NC(=O)Cc3cnco3)C3(CC3)C2)=O)nc(O)n1 80047,N1(C(C2N(C)C(=O)C(F)C2)=O)CCS(=O)(=O)CC1CO 80048,c1(OC)ccccc1CC1CCN(c2ncc(Br)cn2)C1.c12n[nH]cc1NC2=O 80049,C1(NC(CC(C=C)C)=O)CCCCC12CCN(C(=O)C=Cc1cncn1C)CC2 80050,Cc1nc2ncnn2c(C)c1C(=O)N(CC(C)(C)NC(=O)CC1CC(F)(F)C1)C 80051,C(c1cccc(Cl)c1)=CC(=O)NC(CC)CNC(C1CC=CCC1C)=O 80052,N1(c2ccnc(C(=O)OC)n2)CCC(C)(NC(=O)NCCO)CC1 80053,c1(N2C3CC(CNC(C4CCS(=O)(=O)N4)=O)CC2CC3)nc2ccc(Br)cc2s1 80054,CCN=C(NCC(c1ccccc1)N(S(=O)(=O)c1ccccc1)C)N1CCCC1 80055,C(C(=O)NCC1CCC2CC1CO2)(C(C)(C)O)NC(C(N1CCCCC1)C)=O 80056,C1(C(N2CCN(C(c3c(CC)nns3)=O)C(CF)C2)=O)CCCC2(CCC2)C1 80057,N1(C(Cc2n(C)ncc2Cl)=O)CCCCC2C1CCCN2C(=O)C(F)CC1CC1 80058,O=NN1CCCC1C(=O)NCCC1CCN(C(C2CC(CF)C2)=O)CC1 80059,n1(CC)nc(C)c(C(N2CCCC(N(C(=O)CC3(C#N)CCC3)C)C2)=O)c1Cl 80060,c1(NCc2c(C)nc(CC)o2)nccc(=NCC2(OC)CCCC2)[nH]1 80061,c1(C(=O)NCC(CO)NC(C(CC)OC)=O)ccc(N2CCOCC2)cc1 80062,Cc1c(C(=O)NCC2(NC(=O)CCSCC(N)=O)CCCC2)c(C(F)F)nn1C 80063,C#Cc1ccc(C(N2CC3CC3(C(=O)NCC3CC(SC)C3)C2)=O)c(C)c1 80064,N1(C(C2CC(=O)NC2)=O)CCCC(C2(NC(c3c(F)cc(F)cc3Cl)=O)CC2)C1 80065,CC1=NN(C)C(=O)C1CC(=O)NC1CCC12CN(C(=O)Cc1cncs1)C2 80066,n1(C(C)C)cc(C(=O)NC(C)(CNC(C2CC=CC2)=O)C(C)C)c(Br)n1 80067,c1(CC(N2C3CC(NC(c4cc(Br)co4)=O)(C3)C2)=O)ccc2c(c1)OCO2 80068,c1(-c2nc(C3C(CC(C)C)C3)on2)cccc(NC(=O)Cc2cccc(Br)c2)c1 80069,CC(C)S(=O)(=O)CC(=O)N(CC(O)CNC(=O)CNC(c1cccc(O)c1)=O)C 80070,Cc1ccc(C(C)C)c(OC(C)C(N2CC(C)CC2CO)=O)c1 80071,CCC(C)C(O)C(=O)NCc1nc(CNC(c2ncccc2F)=O)cc(O)n1 80072,CCC(C)(C(=O)NCC1CCCN(C(c2ccn(C)c(=O)c2)=O)C1)C(N)=O 80073,c1(CC(c2ccc(F)cc2)(C(=O)O)NCc2cc(Cl)c(Br)s2)cccn2ccnc12 80074,Cc1cnc(C(N2CCC(C(=O)NCCC3CCCCCC3)C(C)C2)=O)c(F)c1 80075,N1(C(c2cnc(CC)s2)=O)CCC(F)(C(=O)Nc2ccc(F)c(C)c2)CC1 80076,CCC(CC(F)F)C(=O)NC1(CNC(C2NC(=O)CC2C)=O)CC1 80077,c1(C(=O)NCC23CC(NC(CC4CC(C)OC4)=O)(C2)C3)cccc2ccn(C)c12 80078,CC(CC(=O)NC(C)(C)CNC(=O)CC1(N2CCCC2)CC1)C1CC1 80079,N1(C(c2ccc(C)cc2)=O)CCC(C(N2CCC(OC3CCC3)CC2)=O)CC1C 80080,c1(C(=O)NC2CCC(NC(C3C(OC)C3)=O)C2)nc(C(F)(F)F)cn1C 80081,c1(C(c2n(CCCCCC)nnn2)NCC2CC(CF)C2)cnn(CC)c1CC 80082,Cc1cc(C(N2CCN(C(C3CCCC(=O)O3)=O)C(CF)C2)=O)nc(O)n1 80083,c1(C(C(=O)NCC2(NC(Cn3c(C)nnn3)=O)CCC2)O)cc(Cl)ccc1F 80084,C(CN1C(=O)Cc2ccccc21)NC(=O)NC1CCCC12CCNCC2 80085,C#Cc1cncc(C(N2CC(OCCNC(C3COCC3C(N)=O)=O)C2)=O)c1 80086,N1(C(CC(=C)Br)=O)CC(NC(=O)CCCN(C)C(C)=O)CC1C 80087,C(=O)(C(O)C(C)(C)CC)N1CC(COC)(CNC(=O)CN2CCC(C)CC2=O)C1 80088,C(=O)(C(F)(F)C1=CCOCC1)N1CC(C2CN(C(CC3CC(=O)NCC3)=O)C2)C1 80089,c1(C(C(=O)NC)N(C2CCC(C(F)(F)F)CC2)C)cc2n(n1)CCCCO2 80090,C1(NC(N)=O)CCN(C(=NCCCC2CCCCO2)NCCF)C1 80091,c1(CC(=O)N(CC(=O)NCC(=O)Nc2ccc(Cl)cc2)C2CCC2)ccccc1C#N 80092,C1(N(C(CCCOCCC)=O)C)CC2CCC(C1)N2C(c1occc1CC)=O 80093,C(CCCC(=O)NCCC(C)NC(c1n[nH]c(C2CC2)c1Br)=O)OCCC=C 80094,O=C(C#CC1CCCOC1)NC1(CNC(c2ccnc(S)c2)=O)CCOC1 80095,c1(NC(C2(F)CC2)C)cc(N2CCCC(CN3CCOCC3)C2)ncn1 80096,CN1CCN(c2nc(Cl)ncc2Cl)C(CNC(C2CC3CCC(C2)S3)=O)C1 80097,C1(F)(CNC(c2ncc(C)s2)=O)CCCN(C(C2(C)CC2C)=O)C1 80098,S(=O)(=O)(c1ccc(N(C)Cc2nncn2C)nc1)N1C(C)C(C(=O)O)CCC1 80099,c1(C(=O)NC2CCN(C(C(CCC)C#N)=O)C2)cnn2c(Br)cccc12 80100,C1(N(C(CC(c2ccc(F)cc2)C)=O)C)CCCCC1N(C(=O)C(N)=O)C 80101,C1(C(=O)NCC(COCC)(C)C)CCN(C(=O)C(C)NC=O)C12CC2 80102,c1(C(N2CC3(C2)CN(C(C2(CF)CC2(F)F)=O)C3)=O)ccc([N+](=O)[O-])cc1 80103,c1(C(=O)NCC23C(CN(C(C(C(=C)Cl)(C)C)=O)C2)C3)cccc2c1ncn2C 80104,C1(C(=O)NC2CN(C(C(C)NS(CC)(=O)=O)=O)C2)(OC)CC(C(F)F)C1 80105,c1(NCC2CCCCN(C(C(c3ccc(C)s3)C)=O)C2)nc(Cl)nc2sccc12 80106,Cc1c(NCCCOCCC(C)C)ncnc1N1CCC(C)(F)C1 80107,c1(C(C)NCC=CC2(C)CCOCC2)cc2ccccc2[nH]1 80108,c1(C(=O)NC2CCCC(NC(CC(C=C)(C)C)=O)C2)cc2ccccc2nc1C 80109,c1(C(=O)NCC2N(C(C(F)=CCC)=O)CCC2)cc2ccc(OC)cc2s1 80110,O=C(CCCCc1ccc(F)cc1)NCCC1CN(C(C2C3CC3C3CC23)=O)C1 80111,C1(NC(C2C(C(C)O)C2)=O)CCCN(C(c2cncn(C)c2=O)=O)CC1 80112,C1(NC(=O)CCc2ccccn2)CCN(C(c2cc(O)nc(Cl)c2)=O)CC1CO 80113,c1(C(=O)NC(CNC(C2C(C)C2)=O)C)nc(C2CC2)ncc1Br 80114,c1(CC(C)C)ncc(C(=O)NC2CC(CCNC(C3CC3C3CC3)=O)C2)s1 80115,c1(NC(c2c(Cl)ccc(Cl)c2O)=O)cc(Cl)cc2nc[nH]c12 80116,C1(C(C)C)C(NC(=O)CCC2CCOC2)CCN1C(=O)CCCN(C)C 80117,c1(C(N2CCN(C(C(CC)C)=O)C(C)C2)=O)oc2ccccc2c1CO 80118,n1(CC)cc(Br)c(C(=O)NC(C)CC(C)NC(c2scnc2Cl)=O)n1 80119,N1(C(c2c(C)nc[nH]2)=O)CC(NC(=O)COC(=O)N(C)C)C2(CCOCC2)C1 80120,C1(C(=O)NCC(N(C)C(c2ccnc(S)c2)=O)C2CC2)CCC2CCC1O2 80121,N1(C(c2n(CC)ncc2)=O)CCCCC(N(C(=O)COCc2ccccc2)C)C1 80122,C1(C(=O)NC2CC(n3cc(C(C)(C)C4CC4)nn3)C2)CCC(C2CC2)C1 80123,C(C)(C)(CN(C(=O)C(C1(C)CC1)NC(=O)C(=O)NCC(F)F)C)OC 80124,c1(OCCOC)cncc(C(=O)NC2CCC(NC(C3CC=CC3)=O)C2)c1 80125,N1(C(CN(C(C)=O)C)=O)CCOC2CN(C(=O)CC3CCSCC3)CC12 80126,N1(C(c2cnc(OC)nc2)=O)C(CNC(c2cc(Br)c[nH]2)=O)CC2COCC12 80127,c1(C(N2C(CCNC(CCOCCOC)=O)CSCC2)=O)cnc2ccoc2c1 80128,c1(C(=O)OC)sc(NC(C2C(O)CCN2Cc2nccn2C)=O)c(C#N)c1C 80129,CC(C)CCC(=O)C(=O)N1CCOC(C(=O)NCC(C)(C)CC(C)O)C1 80130,C1(NC(C(CCC)C)=O)CC(C)CN(C(c2cc(C)cc(Cl)n2)=O)C1 80131,C=CC(C)(CC)C(=O)NC1CCN(C(c2c(C)ccnc2OCC)=O)CC1 80132,C12(CNC(C(CSC)(C)C)=O)CCC(CNC(=O)C3=CSCS3)(CC1)CO2 80133,N1(C(C(C)(C)NC(=O)OC)=O)CCN(C(C)CNC(=O)Cn2ccnc2C)CC1 80134,C#CCCC(O)C(=O)N1CC2CC2(NC(C23CC(F)(C2)C3)=O)C1 80135,Cc1c[nH]c(C(=O)O)c1C(=O)NCCC(C)O 80136,C(=O)(CC(CC(C)C)NC(c1cnc(OC)s1)=O)NC(C#C)(C)C1CC1 80137,CCCCCCC(C)CC(=O)NCCNCC1(O)CCCC(C)C1 80138,N1(C(CSCC(=O)OC(C)(C)C)=O)CCC(C)(NC(C2(C#N)CCCO2)=O)C1 80139,CC(C(C)(C)CO)NC(=O)C(c1cn(C)nn1)NC(=O)CC(C)(C)C1CC1 80140,Cc1ccc(OCc2ccccc2)c(CN2CCN(C)C(C(C)(C)C)C2)c1F 80141,C(CCOCCO)(C(=O)NC(C)C)NC(Cc1c(C)scc1)=O 80142,CCCN=C(NCc1nnnn1C1CC1)NC(c1ccnn1C)COC 80143,C1(CNC(C2CC(=C)C2)=O)CCCCC1C(=O)NCC(Cl)=CCl 80144,C1(C2CN(C(=O)Cc3cn(CC4CCCCNC4=O)nn3)C2)(C(=O)OC)CC1 80145,N1(C(=O)CC2COC3CC2C3)CCC2(CCCN2C(c2cnc[nH]2)=O)C1 80146,n1(C(C)C#N)cccc(NC(=O)C(C)C(N)C2CC2)c1=O 80147,C=Cn1ncc(C(=O)NCC2CCCN2C(=O)CCc2ccc(C)o2)c1N 80148,CC1(CC(=O)N(C2CCN2C(=O)CCCNC(=O)CO)CC(C)(C)C)CC1(Cl)Cl 80149,N1(C(C2CC(OCC)C2)=O)CCCOC(CNC(=O)CCCCC2CCSS2)C1 80150,N1(C(CC(C)(C)Nc2cc3c(cc2)OC(C)C3)=O)Cc2ccnn2CC(CO)C1 80151,c1(C(=O)NCC(CNC(C2CC(C(C)=O)C2(C)C)=O)F)ccc(F)cc1F 80152,N1(C(C2C(C#N)C2)=O)CC(CNC(C2(c3ccc(Cl)cc3)CCC2)=O)C2(CC2)C1 80153,C1(C)(NC(C)=O)CCN(C(=O)CCOC2CN(C(c3sncc3C)=O)C2)C1 80154,N1(c2n(CCOC)c(-c3cnn(C)c3)nn2)CCOC2(CCOC2C)C1 80155,Cn1nc(C(F)F)cc1NC(=O)C(=O)NCCCn1ccccc1=O 80156,C(=O)(C(C)(C)CCSC)N(CCN(C(C(CSC)O)=O)C)C 80157,C(=O)(C1=CCCN(C(=O)COC2CCC3CC23)C1)N1C(C)CC1(C)C 80158,c1(SC)nc(Cl)c(C)c(=NCCN(C)C(C2CCCN(CC(F)F)C2)=O)[nH]1 80159,C1(C(=O)NC2(CNC(=O)COC3CCCOC3)CC2)Cc2ccccc2NC1=O 80160,Cc1ccc(CC(N2CCC(=CC(=O)NCC3CC(F)C3)CC2)=O)nc1 80161,Cc1cc(C(=O)NC2CC(CC(=O)Nc3nccnc3Cl)C2)ncc1[N+](=O)[O-] 80162,CC1CCN(C(=O)C(C)CC(N)=O)C(CNC(=O)Cc2cccc(O)c2)C1 80163,N1(C(C2C(C)C2)=O)CC2CC2(NC(c2coc(Cc3ccccc3)n2)=O)C1 80164,C1(OCC)CCN(C(=NCCNS(C)(=O)=O)NCC(Cl)C(F)(F)F)CC1C 80165,n1(C(C(=O)NCC2CCN(C(C(C=C)O)=O)CC2)C)nc([N+](=O)[O-])cc1C 80166,N1(C(c2cn(C)nc2)=O)CCCC2CCN(C(c3cc(C(N)=O)cs3)=O)CC12 80167,C1(NC(C(N2CC(OCCCCC)C2)=O)=O)CCCC(C(C)CC)C1 80168,N#Cc1cc(NC(C2CN(C(=O)CC3CCCCO3)CCS2)=O)cnc1Cl 80169,C1(NC(CNC(CC(C)C)=O)=O)CC2CC1CC2C(N1CC(C)C(O)C1)=O 80170,Cc1cc(-n2cc(C3CN(C(C4C(C(=O)O)CC4O)=O)C3)nn2)ccc1Cl 80171,C1(C(=O)NCC2C(NC(c3cc(OC)no3)=O)CCC2)CCCC(=O)O1 80172,C(=O)(C(CC1CCCC1)NC(c1ccncn1)=O)NC(C(=O)N(CC)CC)C 80173,C1(O)(CN(C(CCC(C)SC)=O)C)CCCN(C(=O)C(F)=CC2CC2)C1 80174,N1(C(CC(=O)OC)=O)CCCC1C1CCCCN1C(C1CC2(C1)CC(F)(F)C2)=O 80175,N1(C(c2cccnc2)=O)CCN(C(C2CC2(Cl)Cl)=O)C(CF)C1 80176,N1(C(c2cnn(CC(F)F)c2C)C(=O)NCCOC)CCC(OC)C(C)C1 80177,c1(C(=O)Nc2n(CC)ncc2)cc([N+](=O)[O-])ccc1SCC1CC1CC(=O)NC 80178,N1(C(c2nnn(COCC)c2N)=O)CC2(CNC(c3ccsc3)=O)CC1CO2 80179,Cc1cc(NC(c2nncn2C2CCCCC2)=O)ccc1OC(F)(F)F 80180,c1(C(=O)NC(C2CCCO2)CC)ccc(CNC(C2CC(C)(O)C2)=O)o1 80181,CC(CC1CCCC1)N=c1ccnc(NC2CC3CC2OC(=O)N3)[nH]1 80182,N1(C(CC(C=C)CC)=O)CCC(CNC(=O)C2=CCCC2(C)C)C(F)(F)CC1 80183,N(C1CCC(NC(C2CC3CC2C3)=O)c2ccccc21)C(CSC(C)C)=O 80184,C1(C(N(CCOCCCN(C)C(C2(C)COC2)=O)C)=O)CNC(=O)C1 80185,c1(CCNC(C2C(C=C)OCCC2)=O)cccc2cnccc12 80186,c1(C(N2CCCCC2CCCO)C(=O)NC2CCOC2)cc(Cl)ncc1Br 80187,C(=O)(NN=c1ccc2nccn2[nH]1)c1c(C)ccc(C(=O)OC)c1O 80188,c1(CC)cccc(CC(N2CCCC2(C)CNC(=O)Cc2cnn(C)c2)=O)c1 80189,C1(C(N2CCC2(C)CC)=O)(CC)CCCN(C(=O)CCC2CCCOC2)C1 80190,CN(C)S(=O)(=O)NCC(=O)NCCCCC1CCN(C(C2C=CCCC2)=O)CC1 80191,C1(CC)CCCCC1NC(=O)NCC(=O)NC(C)(COC)COC 80192,C1(C)(CCNC(C2(N(C)C(c3nc(Cl)cs3)=O)CC2)=O)CCOCC1 80193,c1(C(=O)NCC2C3CN(C(C(C)OC4CCCC4)=O)CC32)nnn2ccccc12 80194,C1(C(N(CCCC=C)CC)=O)CCOCC1NC(=O)C1=NOCC1 80195,N1(C(CC=C(C)C)=O)CCC(CCNC(=O)C=Cc2cscn2)CC1C 80196,Cc1ccc(C)c(CC(=O)NC2CC(C)N(C(C3CCC(N(C)C)CC3)=O)C2)c1 80197,CCCC(F)C(=O)NCCCOCCC(N1CC(OCC)C(F)C1)=O 80198,n1(CCCC)nnnc1C(c1sccc1Cl)NCC1CC2(CC2)C1 80199,S(=O)(=O)(c1ccc(C(=O)N(C)CCNC(=O)CC2CCC(OC)CC2)o1)NC 80200,Cc1ccc2c(c1)CC(C(=O)NCC(O)CNC(=O)CN1CSCC1=O)O2 80201,N1(C(c2cncc(OCC)c2)=O)CC(C)(C)CCC1CNC(C1(F)CCOC1)=O 80202,N1(C(CC2CC(NC(CCCOCC)=O)C2)=O)CCOCC(O)C1 80203,N1(C(C(CC=CC)C)=O)CCC2(CC1)CN(C(c1cccc(CO)c1C)=O)C2 80204,c1(C(c2nn[nH]n2)CNC(CNC(C)(C)CO)=O)ccccc1F 80205,O=C(C1CCCc2n[nH]cc21)NC1(CF)CCN(C(=O)C(F)(F)C2(O)CCC2)C1 80206,c1(C(=O)NC(C(C(C)C)NC(=O)CSS(C)(=O)=O)C)cncc2nc(O)[nH]c12 80207,NS(=O)(=O)c1n[nH]cc1C(N1CCCC(NC(=O)CC2CC(=O)NC2=O)CC1)=O 80208,Cc1cnc2cc(C(N3CCOCC3CNC(=O)CCc3csnn3)=O)ccn12 80209,C(=O)(C1=CC2(CN(C(=O)C(C(CC)CC)OC)C2)OC1)N(CCC#C)CC 80210,C(=O)(C(CNC(=O)C(OC)OC)C(C)C)Nc1c(CC)noc1C 80211,C1(C(=O)NCc2cc(COC)n[nH]2)CCCN(C(=O)COCCC(C)C)C1 80212,c1(CNC(COC(CC)(C)C)=O)cn(CCNC(=O)CC2(C)CCCO2)nn1 80213,Cc1cc(C#N)ccc1N(C1CCN(c2ncc(Br)cn2)C1)CC(F)(F)F 80214,C12(C(N(CCN(C)C(c3cnc(O)s3)=O)C)=O)CCC(CC1)C2(C)C 80215,c1(C2OCCN(C(C(CCOC(CC(C)C)=O)F)=O)C2)ccc2ccccc2c1 80216,C1(C(=O)NC)CCC2(CCN(C(C3CC(F)(F)C3)=O)CC2)O1 80217,Cc1cccc(Oc2ccc(NC(=O)COc3c(C(=O)NC)cccn3)cc2)c1 80218,c1(C(N2CCC(c3ccncn3)CC2)C(=O)NC(C)C)cccc2cn(C)nc12 80219,CC1(C)OCCC1C(=O)NC1CCC(NC(C2CC(C)(C(C)(C)C)C2)=O)CC1 80220,C(CCCCCNC(C1(C)CCCCC1)=O)NC(C(C)Cc1ccncc1)=O 80221,c1(-c2nccc(C(=O)NC)c2)ccc(F)c(C(N2CCC(CC(=O)NC)C2)=O)c1 80222,C(=O)(C1=CC2(CCN(C(=O)Cc3ccoc3)C2)C1)NCC(N1CCOCC1)C 80223,C(=O)(CC(CC)C(C)(C)C)NCCN(CCCCCC)C(=O)C(O)CC1CC1 80224,C(C(=O)NCCC1(CNC(=O)CCc2nccs2)CCC1)(c1cccs1)SC 80225,C=CC(C)(C)CC(=O)NCCN(C1CCCC1)C(=O)COCC1(F)CC1 80226,c1(C(=O)NC2CCC(CNC(C3(SCC)CC3)=O)C2)cncc2c[nH]nc12 80227,C1(NC(C(C(C)C)O)=O)C2CC1CN(C(c1cc(C#N)c[nH]1)=O)C2 80228,N1(C(C(c2cccnc2)NC(C2CC(C)=C(C)CC2)=O)=O)CC2CCCC(C2)C1 80229,N1(C(C(C(C)C)SC)=O)CCCC2(C1)CN(C(c1cccc(O)c1F)=O)CCO2 80230,C12(C(=O)NC3CCN(C(c4n[nH]c(C)c4Cl)=O)C3)CCCN(CC1)C2 80231,CC1(CNC(c2cc(N)ccc2O)=O)CCCN(C(c2c(F)ccnc2Cl)=O)C1 80232,CC1(C)CN(C(c2cc(C3CC3)no2)=O)C(CNC(C2CCCOC2)=O)CO1 80233,c1(C(=O)NCC(C)(C2CCC2)NC(=O)CCCC#N)cc2cncn2c(O)n1 80234,c1(C(N(C2CCN(C(CC(C=C)C)=O)C2)CC)=O)cc2nc(Cl)ccc2s1 80235,c1(CCOC(C)C)nc(-c2cnc[nH]2)n(-c2nccn2C)n1 80236,C1(NC(CC(CC)C)=O)CCOC12CCN(C(=O)C(C)OC)CC2 80237,C1(NC(c2cc(COC)on2)=O)CC1C1CCN(C(=O)Cc2sccc2C)CC1 80238,c1(C(CO)NC(NNC(c2cccc(OC)c2)=O)=O)ccc(S(C)(=O)=O)cc1 80239,c1(C(=O)NC2CC(NC(C34C=CC(CC3)C4)=O)C2)c[nH]c2ccc([N+](=O)[O-])cc12 80240,C1(C(=O)NCCCN(C(c2cncc(N(C)C)n2)=O)CC)CCCCC1C1CC1 80241,N1(C(CC(CC)NC(=O)CCN2CCOCC2)=O)CCC(O)C(CO)C1 80242,Cc1nc(C(C)C)ccc1C(=O)NC1CN(C(=O)CN2CCC(C)CC2)CC1F 80243,C(=O)(C(C)(C)CS(N)(=O)=O)NC1CC(C)(C)N(C(=O)CC(F)(F)F)C1 80244,Cc1ccc(O)c(C(N2CCC(C(F)C(=O)NCC=Cc3cccnc3)C2)=O)c1 80245,c1(OC)ccc(C(=O)NCC2CC(NC(C3(n4cncn4)CC3)=O)CCO2)cc1 80246,C1(COC)COCCN(C(=O)CC(C)NC(c2cc(Br)cs2)=O)C1 80247,C(=O)(C1CCc2cc(C)ccc21)NCC1(NC(C(CC(CC)CC)F)=O)CCC1 80248,C(CC(=O)NOCC1CCCO1)C1CCN(C(C2(COC)CCCC2)=O)C1 80249,c1(CC(=O)NC2CCC(NC(C3CCCC3CF)=O)C2)c[nH]c2ncccc12 80250,O(NC(=O)C(CCF)NC(c1cccc(O)c1F)=O)CCCC=C 80251,c1(C(=O)NC2CCCN(C(CC3(C=C)CCC3)=O)CC2)cc(C)cc(OC)c1C 80252,N1(C(c2[nH]cc(C)c2)=O)CCC2(C1)CN(C(=O)CCCNS(C)(=O)=O)C2 80253,c1(OC)ccc(C(=O)NC(C2(O)CN(C(C3CCCSS3)=O)C2)C)cn1 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80863,O=C(CCCN1CCCC1)NC(C(=O)NCC(F)C1CCC1)c1ccoc1 80864,C1(CNC(C(C)=C(CC)C)=O)COC(C)(C)CN1C(C1CCCCC1)=O 80865,C1(CNC(C2C(C)(C(F)(F)F)C2)=O)CC2CCC1N(C(C1(CO)CCCC1)=O)C2 80866,N(C(=NCCC1COC(C)(C)OC1)NCC(N1CCOCC1)C)CC(=O)NCC 80867,Cc1nc(O)ccc1C(=O)N(C1CCCN(C(=O)COCP(C)(C)=O)CC1)C 80868,Cc1ccc(CO)cc1NC(=O)CCC1CC(NC(c2cccn2C(C)C)=O)C1 80869,C(=O)(C1Cc2ccccc21)N1CC(NC(c2coc3c2COC3)=O)C(O)C1 80870,C(N=C(NC1CC1)N1CCC2=C(COC2=O)C1)C1CN(C)C(C)(C)C1 80871,CC(CCC(=O)NC1CN(C(C2CC2Br)=O)C1)N(C)C 80872,CC1(CNC(=O)CCCC#N)CCN(C(=O)COCC2CCCO2)CC1 80873,C1(C(=O)NCCNC2CCCCC2)CCCC(Nc2cn[nH]c2)C1 80874,CC(O)CCCCCC(=O)NCCN(C)C(c1c(F)cc(C(F)(F)F)cc1F)=O 80875,C1(NC(C2CC(OCC)C2)=O)CN(C(=O)Cc2csc(-c3ccco3)n2)CC1C 80876,c1(CNC(=O)NC(CC(=O)OC)CC(C)C)cccc2nc(CO)[nH]c12 80877,C12(NC(Cc3cc(CC)no3)=O)CCCN(C(=O)CSc3cnn(C)c3)CC1C2 80878,c1(C(N2C(C)CC(NC(c3cccc(COC)c3)=O)C2)=O)cnn2c1CCCC2 80879,N1(C(C(=O)NCc2ccc(C)o2)C)C(C)CCCC1C 80880,S(=O)(=O)(c1cccc(C(=O)OC(C)(C)C)c1)N(C1CCCCCC1O)C 80881,C1(CCNC(c2nn(CC)c(C3CC3)c2)=O)CCCN(C(=O)C(N)=O)CC1 80882,c1(N(C)CC2CCN(CCC#C)C2)ccc2c(n1)CCC2=O 80883,C1(CC=C)(NC(=O)Cc2cnc(C)o2)CCCN(c2cc(C)nc(SC)n2)C1 80884,N1(C(CCC(C)N(C)C)=O)CC(CO)C2(C1)CN(C(C1CC=CC1)=O)C2 80885,CCC(CCCC(=O)N1CCCC1CN(C)C)NC(C1CC(O)C(F)C1)=O 80886,Cc1oc(C(C)C)cc1C(=O)NC1CCOCC1NC(=O)CCc1cc[nH]n1 80887,C1(CN(C(c2c(C(C)C)con2)=O)C)COCCN1C(=O)C(O)CCN(C)C 80888,C(=O)(C(CC)C(=O)N1CC=C(CNC(c2cccc(CO)c2)=O)CC1)OC 80889,N1(C(c2nnn(C(C)(C)C)n2)=O)CCC(C(F)(F)F)C(NC(=O)C(F)C2CC2)C1 80890,C1(C(N2CC(CN(C(=O)COCC3(F)CC3)C)OCC2)=O)Cc2cscc2C1 80891,c1(C(=O)OC)cc(NC(Cc2ccccc2OC(C)C)C(C)C)ccc1C 80892,N1(C(C(C(C)C)n2cncn2)=O)CCC(CO)(NC(=O)CCCCC#N)CC1 80893,C(CC(F)(F)Cn1cc(-c2conc2C(F)(F)F)nn1)NC(C1CCCCO1)=O 80894,N1(C(c2c(C)nn(C)c2)=O)CCN(C(c2cc(C(C)C)ccc2F)=O)C(CF)C1 80895,c1(OC)ccc(Br)c(OC)c1NC(C1CC(=O)N(C)C1c1ccccc1)=O 80896,C1(C(N2C(CC)C(NC(=O)CC(F)(F)F)CC2)=O)CCCCCC1(F)F 80897,Cc1nn(C2CCC2)cc1C(N1CC2CC1C2NC(=O)Cc1ccnn1C)=O 80898,Cc1cccc(C)c1C(N1CC(NC(c2cc3sccc3[nH]2)=O)C2(CC2)C1)=O 80899,C1(C(N2CCC(CCC)(CO)C2)=O)CC(C)CN(C(c2cccs2)=O)C1 80900,C1(C(N2C(CC)CCC2)=O)COC2(C1)CN(C(C1(C(=O)N(C)C)CC1)=O)C2 80901,C1(NC(c2cc(C)c(C(C)C)cc2)=O)CCSC12CN(C(C1CC13CC3)=O)C2 80902,c1(CC(C(N2CC(C#N)(SC)C2)=O)C)ccc(F)c(F)c1 80903,C1(C(=O)NCc2ncc(C)s2)CC2(CCN1C(C1CC(C)CCO1)=O)CC2 80904,c1(OC)cnc2c(c1)C(NC1(CO)CC(OC)C(OC)C1)CCN2 80905,C(C(=O)NCC(O)CNC(=O)C(OC)OC)(OCC)OCC 80906,CC#CCCCC(=O)N(CCCOCCN(C)C(C12CCCC1(C(N)=O)C2)=O)C 80907,c1(CNC(c2c(Br)ccnc2Cl)=O)c[nH]c2cccnc12.C12CN(C1)C2 80908,C1(NC(c2c(CC)nns2)=O)CCC(C)N(C(C2(COC)CCC2)=O)C1 80909,CCC(CN(C)C)C(=O)N1CCC=CC1C(=O)N(CC(O)CF)C 80910,C1(CNC(C(C)Oc2ccccn2)=O)C2CN(CCC3CC3)CC12 80911,c1(C(=O)NC2C(NC(c3c(C)nc(Br)o3)=O)CC2)cnc2ccccn12 80912,C1(CNC(c2cc(C)c(Cl)cn2)=O)C(C2CC2)CCN1C(=O)CCc1cnco1 80913,C1(CC(N2CC(C(C(=O)NC(C3CCCCC3)COC)OC)C2)=O)CCCN(C)C1 80914,C1(C(N2CC(C(N)=O)(CNC(C3CCC(=O)N3)=O)C2)=O)CC2C=CC1O2 80915,C1(CCC)CCC(C(C(=O)NC(C)CC)N(c2ccncc2)CC)CC1 80916,N1(Cc2ncc(C)s2)CCN(CC(c2ccccc2)O)CC1 80917,N1(C(C(C)(C)C2CCN(C(c3cc4n(n3)CCO4)=O)C2)=O)CCC2(CC1)CSC2 80918,C1(CC(=O)NCCOCCCNC(C2CC(CC)C2)=O)CCCC2CCCCC12 80919,C1(NC(CC2(CC)CCC2)=O)C=CC(CC(=O)NC(C(O)CO)C2CC2)C1 80920,C1(C(=O)NC(C2(O)CN(C(c3cc(N(C)C)ccn3)=O)C2)C)CC(C2CC2)=NO1 80921,C(=O)(C(C)C(F)(F)F)NCC=C1CCN(C(c2cncc(CC)c2)=O)CC1 80922,C(=O)(C1=CC(C)(CC)C1)NC(C1(O)CN(C(c2c(CCC)[nH]cc2)=O)C1)C 80923,N1(C(C(C=C=C)C)=O)CCOC2(C1)CN(C(=O)C(C)(C)CC1CCOCC1)C2 80924,CC(CC(=O)N1CC2(CNC(c3ccc4nnnn4c3)=O)CC1CO2)C(C)(C)C 80925,c1(C(=O)NCC(C(C)C)N(CCC)C)cccc(OCC2C3COCC23)c1 80926,C(=O)(C1CCc2cccc(=O)n21)N1C(C(=O)NC)CC(OC)C1 80927,c1(C(=O)NC2CC(N)C2)cc(N2CCOCC2)nc(Cl)c1 80928,C1(NC(C23N(C(C4N(CC)CCC4)=O)CC(C2)C3)=O)CCCCCCC1O 80929,Cc1c(Br)cc(S(=O)(=O)N2CCCN(Cc3ccccc3)C(C)C2)c(C)c1C(=O)O 80930,c1(C(=O)NC2(C(=O)NCC(O)CC(F)(F)F)CCCCC2)cccn2nccc12 80931,N1(C(CNC(=O)OC)=O)CCC(NC(c2ncc3[nH]ncc3n2)=O)C2(CCC2)C1 80932,CC(C)(CC(F)C(=O)NCc1nc(C2CC2)n[nH]1)NC(c1cccc[n+]1[O-])=O 80933,N1(C(c2c(OC)ncc(Br)c2)C(=O)NC2CCOC2)CCCC2C(O)CC12 80934,Cc1nn(C)c(C(C(=O)NC2CC2)N(C)CCC2CCCCN2C)c1Br 80935,N1(C(C(C)OCCC(C)C)=O)CCC(C(C)C(=O)NCC2(C)CCCO2)CC1 80936,C12(C(=O)NCCCN(OC)C)CCCC1CCN2C(C1CCCOC1)=O 80937,N1(C(C2(CCCF)CC2)=O)CCC(O)(c2ccccn2)CC1 80938,CC1(C)CC(C(=O)NCC2(C)CC2(F)F)CN1C(c1ccc(C#N)cn1)=O 80939,N1(C(C=C(CC)CC)=O)CCC(NC(=O)CC2CC2(C)C)C12CCC2 80940,c1(OCC(=O)NC2C(NC(c3c(CC)c[nH]n3)=O)C2)nn(C)cc1[N+](=O)[O-] 80941,C1(CC(=O)N(CCCNC(=O)C(c2ccc(C)s2)C)C)(CC)CCOCC1 80942,C#CCC(CC(F)F)C(=O)N1CC(NC(c2n[nH]c(C)n2)=O)CC1(C)CC 80943,C(=O)(C1=NNC(=O)C1)N1C(CNC(=O)CC2C=CCC2)CC1 80944,Cn1ccnc1C(F)(F)C(=O)NCC1CCN(C(=O)Cc2cnc[nH]2)C1 80945,c1(OCC)cnc(N2CC3C(CNC(=O)C(C)CCN(C)C)C3C2)nc1C 80946,C(c1cccnc1)=CCNC(C(c1ccco1)NC(=O)CC1CC1)=O 80947,Cc1ccc(C(F)(F)C(=O)NC2CN(CC(C)C)C2)cn1.C12CC1CNC2=O 80948,C(=O)(C(C)(C)C(C)NC(c1cn(C2CC2)cn1)=O)NCC(N1CCCC1)C 80949,c1(OC)cn(CC(=O)NCCCC(C)(C)NC(=O)COC(=O)CO)c(C)cc1=O 80950,C(=O)(CC(C(F)F)NC(c1cccc(OC)c1)=O)NC(CC)(C)CO 80951,N1(c2n(C3CCC(C)C3)c(-c3ccccn3)nn2)CCn2nnnc2C1 80952,C1(NC(c2cc(C)c(C)o2)=O)CC2CC(C1)N(C(=O)CCc1cn(C)nn1)C2 80953,C1(NC(Cc2c(C)cc(F)cc2)=O)C2COCC1CN(C(=O)CC1CC(F)C1)C2 80954,C1(C(=O)NC2CCCN(C(C3(C4(C)CC4)CC3)=O)C2)CCC2CC1CO2 80955,n1(CC(=O)NC(C)C(C)NC(=O)COC2CC=CC2)ccnn1.C(C)(C)C 80956,CC1CN(C(=O)C(c2ccccc2)O)CC1CNC(=O)C(c1ccccc1F)O 80957,c1(C(=O)NC2CCCC(N(C(=O)CC(C)(F)F)C)C2)cc(S(C)(=O)=O)cnc1O 80958,C(=O)(CCN=c1[nH]ccs1)N1CCC(CNC(C(CC)Cc2ccccc2)=O)C1 80959,c1(C(N2C(CNC(c3ccnc4cc[nH]c34)=O)CCC2)=O)cc([N+](=O)[O-])ccn1 80960,c1(C(=O)NCCC2CCN(C(CCC3CCN(C)C3)=O)C2)ccnc2ccnn12 80961,C1(C(=O)NCCCN(C(=O)CCc2ccoc2)CC)CCn2ncnc2C1 80962,C1(C(=O)Nc2cccc(C)c2)CC2(CCN1C(=O)CNC=O)CC2 80963,N1(C(Cc2n(C)ncc2Cl)=O)CC(CNC(C2CCCC(=O)N2)=O)C2(CCC2)C1 80964,CCCCC(C(=O)N1CC2CN(C(c3ccc(CO)cn3)=O)CC2(C)C1)C(C)C 80965,c1(OC)ccc(O)cc1C(N1CC(OC)CC1CNC(=O)CC12CCCC1C2)=O 80966,N1(C(C(C2CC2)OC)=O)CC(O)CC1CC(=O)NC(C1CCOC1)CO 80967,c1(C(=O)NC)ccc(CC(=O)NC2C=CCN(C(=O)CSCC#N)C2)cc1 80968,C#Cc1cccc(CCC(=O)NC2CC23CC(NC(=O)COCC(F)F)C3)c1 80969,N1(C(C2(SC)CCC2)=O)CCN(C(C2CC(C#N)C2)=O)C2CCCCC2C1 80970,CC1CN(C(C2(CCNC(C3(O)CCCCC3)=O)CCCC2)=O)CC1NCCO 80971,c1(OC)cc(Cl)c(Br)cc1NC(c1ccc(-c2csc(C)n2)cc1)=O 80972,c1(C(N(C2CCN(c3ccc(C)cc3)CC2)C(CC)CC)=O)c(C)n[nH]c1C 80973,C1(C(=O)NC(C)CC(C)NC(=O)C2CC2)CC2(CCC(F)(F)CC2)CO1 80974,Cc1csc(=O)n1CC(=O)NCC1(CNC(C2CCC(=O)O2)=O)CCCCC1 80975,C(CCC(C)(C)SC)NC(C1(COC)CN(C(=O)CSC(F)(F)F)C1)=O 80976,c1(C(=O)NC(CC(C)C)(C)CNC(=O)CC2CCC2)cnc2n1CCCC2 80977,Cc1cc(C(=O)NC2CN(C(=O)CC(C)c3ccncc3)CCC2F)cc(F)c1 80978,C1(NC(C2(C(=O)NC)CCC2)=O)CCN(C(=O)Cc2csnc2C)CC1C(C)C 80979,C(=O)(C(CNC(=O)CSC(C)C)CCC)NCCC#CCC 80980,N1(C(C=CCOC)=O)CCCC(C(=O)NC(C)C(N)=O)C1 80981,c1(COC)cccc2sc(NC(C3CCC(C#N)C3)=O)nc12 80982,c1(SCC(=O)NCC2CC(F)(CNC(CCCOC)=O)C2)cc(C)ccc1C 80983,c1(C(N(C(C)CCO)C)=O)ccc(C2COCCN2C(C2CC2C(F)F)=O)n1C 80984,c1(CCNC(N2C(C(N)=O)CC(O)C2)=O)c[nH]c2c(F)cc(Cl)cc12 80985,C12(CNC(CSCC#C)=O)CN(C(c3sccc3C#N)=O)CC1CCO2 80986,C(=O)(C(C)(C)C(=O)NN1C(=O)C(C)N(C)C1=O)Nc1nnc(C(CC)C)s1 80987,C1(NC(CCCn2c(C)ncc2)=O)CC(C)N(C(C2CN(C3CCOC3)C2)=O)C1 80988,CCCC(C)(C)C(=O)NCC1(F)CCN(C(c2noc(C3CC3)c2C)=O)C1 80989,C12(CNC(C3C(C)(C)CO3)=O)CC1CN(C(c1cnc(CC3CC3)s1)=O)C2 80990,C1(C(=O)OC)CCC(Cn2cc(CNC(c3cn(C)nc3Cl)=O)nn2)CC1 80991,CC1(C(N2CCOC(CNC(=O)Cn3cc(C4CC4)cn3)C2)=O)CC2CC2C1 80992,C(c1cccc(F)c1)=CCC(=O)N(CCN(C(C1CC2(CC2)CO1)=O)CC)CC 80993,Cc1ccc(-c2cc(F)ccc2CO)c2nc(C(=O)NCc3ccc[nH]3)cn12 80994,N1(C(CNC(C2C(C)=CCS2)=O)=O)CC2CCCCCC2C1 80995,Cc1ccc(CC(N2CCCC2(CO)CNC(=O)CN(C)C)=O)cc1Cl 80996,c1(COC)nn(C)c(Cl)c1C(N1CCCCC(N(C(=O)C=CCO)C)C1)=O 80997,c1(C(N2CCCC(NC(COC(CC)(C)C)=O)C2C)=O)cnc(S(C)(=O)=O)s1 80998,c1(C(=O)NCC2CN(C(CNC(C(CC)C)=O)=O)CC2C)cc(C)c(F)c(C)c1 80999,CC1CN(C(=O)COC2CCCC(C)C2)CC1NC(=O)C(N1CCCCCC1)C 81000,c1(NC(C2C3CN(C(C(CC=CC)C)=O)C2C3)=O)cnc(C)nc1C 81001,C1(OC)(CNC(C2SCCS2)=O)CCN(C(=O)Cc2cccc(Cl)c2)C1 81002,N1(C(C(C)SCC)=O)CC(CO)C2(C1)CN(C(=O)C(c1cnn(C)c1)O)C2 81003,N1(C(Cc2c(C)cccn2)=O)CC2CCC1C(NC(c1cc(N)ccc1F)=O)C2 81004,C1(NC(C2(NC(CC3(C)CC3)=O)CCSC2)=O)CC2(CCOC2)C1 81005,Cc1noc(C)c1CSCC(=O)N(CC(C)NC(C1(O)CCOCC1)=O)C 81006,C=CCCC(C(=O)N1CC(c2nncs2)C1)NC(=O)C(C)CCCC 81007,C(=O)(CCCC(=O)N1CC(C2CC2)(C(=O)NC2(C)CCSC2)C1)OC 81008,C12(NC3CN(CC(N)=O)C3)CC(c3nn[nH]n3)(C1)C2(F)F 81009,c1(CCC(=O)OCC)ccc2c(n1)N(C(=O)NCC1CCCCC1)CCC2 81010,CC1(C)OC2(C(=O)NCCCn3cc(C4(O)CCC4)nn3)CCC1C2 81011,C1(CC(=O)OCC2CN(C(=O)OC(C)(C)C)C2)CCCCNCC1 81012,c1(C(=O)NCC2CC(NC(C(CC(=C)C)C)=O)C2)cc2ccc(F)cc2o1 81013,C1(NC(=O)C2=NOC3COCC23)CCC2(CCCCC2)CC1 81014,n1(CC(=O)NCC2C=CCN2C(=O)CC2C=CCC2)nc(C(F)F)c2c1CCC2 81015,c1(C(=O)NCC(CNC(c2ccc(Cl)c(Cl)c2)=O)F)cccc2ccncc12 81016,CC1CC(C(=O)NCC(C)(C2CC2)NC(c2cc(O)nn2C)=O)CCC1C 81017,c1(OCC(=O)OC(C(=O)Nc2c(N)cc(C)c(F)c2)=O)ccc(S(N)(=O)=O)cc1 81018,C1(C(=O)NC2CCC(C)(CNC(c3nnc(C)s3)=O)CC2)CN2CCN1CC2C 81019,CCC(CC)(C(=O)NC(CNC(C1CCCC(C(N)=O)C1)=O)C(C)C)OC 81020,C=C1CC(C)(NC(=O)CC2C(NC(=O)CC3CC(C)C3)CC2O)C1 81021,C1(NC(CCC=C=C)=O)CN(C(=O)C(Cl)=CCl)CC2(CC2)C1 81022,CCC(F)(F)CC(=O)NC(C)(CNC(C1CC(OC)C1)=O)C1CCC1 81023,C(=O)(CCC(F)(F)C(=O)N1CC(C)(C)CC1CNC(=O)CC(C)(C)CC)OCC 81024,C12(C(=O)N)CCC(CO)(CC1)C2.C(=O)(CCNC(C1CC(CO)C1)=O)NC(CC)C 81025,c1(C(=O)NCC2(OCC)CN(C(=O)C(C3CCC(=O)N3)C)C2)ccc(=N)[nH]c1Cl 81026,c1(C(=O)NC(CC(C)NC(Cc2c(C)cccc2)=O)C)ccn(C(C)C)c(=O)c1 81027,C12(C(=O)NCC3C(CNC(C4(CC#C)CCCC4)=O)C3)CCCC(CO1)C2 81028,C(=O)(C(C)CNC(C1CCOCC1)=O)NCCOCC 81029,C(c1cc2ccccc2o1)=CC(=O)NCc1cc(Cl)ccc1OCCO 81030,c1(CCC(=O)NC2CCC2NC(=O)C=CCOc2ccccc2)ccccc1F 81031,C1(C(=O)NCCN(CCC)C(C2CCNC2=O)=O)COCCC1(F)F 81032,C(=O)(C(O)C(C)C)NC1CC(C(=O)N(C)Cc2ccc(C3C(C)C3)o2)C1 81033,C1(C(N(C)CCNC(=O)Cc2ccccc2O)=O)CN2CCC1(C)CC2 81034,C(CO)(CCCNC(c1coc(C)c1)=O)NC(C(CSC)OC)=O 81035,CC#CCC(C(=O)N1CCCC1CCO)NC(c1ccc(CC)nc1)=O 81036,c1(C(N2CCC(SC(C)(C)C)CC2)=O)ccc(N)cc1[N+](=O)[O-] 81037,Cc1ncn(C)c(=O)c1C(=O)NCC1(NC(=O)Cc2ccsc2Cl)CCC1 81038,C1(C(=O)NC(C)CCNC(C2(C(C)(F)F)CCC2)=O)CCOC2(CCCC2)C1 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81093,CC1CN(C(=O)CCN(C)C(C2C3CCCCC23)=O)CC1O 81094,Cc1cccc(C)c1C(N1CCC1CNC(C1(F)CCOC1C)=O)=O 81095,c1(C(=O)NC2C(CC)N(C(C3COC(C)C3)=O)CCC2)ccc(Cl)c(Cl)c1N 81096,C1(C(=O)NCC2(OC)CN(C(C3COC(=O)N3C)=O)C2)CC(C)CC(C)C1 81097,c1(CC(N2CC(C)(C(=O)Nc3cnc(Br)cn3)C2)=O)ccc2c(c1)CCCO2 81098,c1(OCCC)cccc(CC(=O)NCC2CCN(C(C34CCC(C3)C4)=O)C2)c1 81099,C(C(C)CC(=O)N1CCC(N(C(c2cn(C)cc2C)=O)CC2CC2)C1)OC 81100,c1(C(N(CC)CC2CCCN2C(=O)C=CC(C)(C)C)=O)ccc(N(C)CC)cc1 81101,C1(C(=O)NCC(CNC(c2cnc(OC)nc2C)=O)O)CCC(=C(F)F)CC1 81102,N1(C(c2cc(OC)ncn2)=O)CCC2(CCC(NC(C3CCC(O)CC3)=O)C2)C1 81103,C12(C(=O)NCC(C)CNC(=O)C3=NOC(C)C3)CC(C)(C1)OC21CCC1 81104,N1(c2c(C#N)cnc(SC)n2)CCC2(CCC2NC(C2CC=CCC2)=O)CC1 81105,CC1CN(C(C2CCN(C(C3CC(O)CN3)=O)CC2)c2ccccc2)CC(C)O1 81106,N1(C(c2c(C)cno2)=O)CCCC(N(C)C(c2ccc(-c3ncc[nH]3)nc2)=O)C1 81107,c1(C(N2CC(CNC(C3(C)CC(=C)C3)=O)C(C)C2)=O)cc(C)nc2cc(C)nn12 81108,c1(OC)ccc(C(=O)N(C2CCCC2)CCNC(c2ccccn2)=O)nc1Cl 81109,Cn1nnc2cc(C(=O)NCC3CC3CNC(c3conc3C(C)(C)C)=O)sc12 81110,c1(OC)nc(Cl)ccc1C(=O)NCC1CC(CNC(=O)C2CC2)CO1 81111,c1(C(=O)NC2CC(OC)CN(C(=O)C(C)(C)N(C)C)C2)cc2ccc(C)cn2c1 81112,N1(C(C=CCC)=O)CCC2(C1)CN(C(=O)CCCc1n[nH]c(=N)s1)CCO2 81113,c1(C(C)(F)F)cncc(C(=O)NC2CCCCC2NC(=O)CCC2CCCO2)c1 81114,Cn1nnc2cc(C(=O)NC3CCC34CN(C(c3cc(Cl)cs3)=O)C4)cnc12 81115,C1(N(C)C)(C(=O)NCC(O)CNC(=O)CCC2CCCO2)CCCOC1 81116,C1(C(N(C(CCO)C(C)(C)C)C)=O)N(C(=O)OC(C)(C)C)CC12CCCC2 81117,N1(C(C2CCN(C(C(C)OCCN(C)C)=O)C23CCC3)=O)CCC2(COC(=O)N2)C1 81118,C1(C(C)(C)NC(CC2CC(=C)C2)=O)CC2CCC(C1)N2C(c1c[nH]c(=N)s1)=O 81119,c1(C(N2CCC(C(C)NC(=O)C(C)=CC(C)(C)C)C2)=O)ccccc1S(C)(=O)=O 81120,C1(CCC(=O)NC(C)CN(C)C(c2nnnn2-c2ccccc2)C)CCC(=O)N1 81121,c12cc(nc(=O)[nH]1)NN2C.c1(CCCN(C)C2CC2)ccc(Br)c(F)c1 81122,CCC(C)(CCC(C)C)C(=O)NC1CC(C)(NC(=O)C(C)S(=O)(=O)C(C)C)C1 81123,c1(CN(C(C(=O)NCCSC)CC2CCCCC2)C)ccc(F)cc1Cl 81124,C1(NC(CN(CCC)C)=O)CCN(C)C12CCCN(C(=O)CC1CCCCO1)C2 81125,C(N=c1[nH]ncs1)C1C(NC(C2CCN2Cc2ccccc2)=O)CCC1 81126,C=CC1CN(C(=O)C(CC(F)F)N(C(=O)C(CCC)OCC)C)CCO1 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81145,N1(c2cc(N3CCCC(c4n(C)ccn4)C3)ncn2)CC2C3CCC(CC3)C2C1 81146,C1(NC(C2(OCC)CCC2)=O)CN(C(c2cnc(C3CC3)nc2)=O)CC1C 81147,C(=O)(C1=CCC(C(F)(F)F)OC1)NC(C)CCN(C)C(c1cnc(S)nc1)=O 81148,C1(C(=O)NC2C3CN(C(=O)Cn4cc(Cl)cn4)CC23)CCC=CCCC1 81149,c1(C(=O)NC(C)(C)CN2CCCCC2=O)cnn2cc(F)cc(F)c12 81150,C1(NC(c2c(C(C)C)cccc2)=O)CN(C(C2(C)CC2(F)F)=O)CC1S(C)(=O)=O 81151,c1(C2C(C(=O)NCCC3(O)CN(C(C(CC)F)=O)C3)CC2)ccc(Cl)cc1F 81152,C(CCCCC(=O)NC1(C)CCN(C(=O)C(C)Cc2cnn(C)c2)C1)OC 81153,N1(C(CN(c2ccc(OC#N)c(O)c2)C)=O)CCN(Cc2ccccc2)C2CC12 81154,C12(C(N3CCC(C(C#C)C)CC3)=O)CCN(C(=O)CCC=C(C)C)CCC1C2 81155,C1(NC(c2ccc(C3CC3)s2)=O)CCCC12CN(C(=O)COCC1CCOC1)C2 81156,c1(C(=O)NC(CNC(CC(CCC)O)=O)C2CCC2)c(F)cc(F)c(O)c1F 81157,C1(NC(C(C)CF)=O)CN(C(c2cc[nH]n2)=O)C2(CCOCC2)C1 81158,c1(C(=O)NCCNC(=O)COCC2CCOC2)c[nH]nc1C(F)(F)F 81159,Cc1cccc(Cn2nc(-c3ccc(C(F)F)cn3)nc2-c2ccsc2CO)c1 81160,c1(C(=O)NC2C(NC(=O)COC3CCCC3)CC2)cc(C2CCCCC2)no1 81161,O(NC(=O)C(c1cccnc1)NC(=O)Cc1cn[nH]c1)CC1(C)CC1 81162,c1(C(=O)NC(CCCNC(C2(C)CCC(OC)CC2)=O)C)ccc(C#N)c(C)c1 81163,CCCCCCCCC(=O)N1CC2(CC(NC(c3cc(Br)cnc3C)=O)C2)C1 81164,C1(C(=O)NC2(C(F)F)CC(C(=O)NC3CN(C(=O)OC)C3)C2)CC(C)(C)CO1 81165,C=CCCCN=c1[nH]cnc(Cl)c1C1CC1.C(=O)OC 81166,CC1(C)CC(CC(=O)NCC2(CCNC(=O)CCCc3ccsc3)CC2)CCO1 81167,Nc1cc(C(=O)NCC2CN(C(c3cccs3)=O)CC2C(F)(F)F)ncc1Cl 81168,C=CC(C)(C)CC(=O)NCC1CN(C(=O)C(C)=C(C)CC)CCC1C 81169,C(=O)(C1=CCCC1(C)C)N1CCC(C(CNC(c2ccc(C#C)cn2)=O)F)CC1 81170,c1(C(=O)OC)ccccc1CC(C)(CO)n1cc(-c2cc[nH]c(=N)c2)nn1 81171,N1(Cc2ccc(C)c(Cl)c2)CCNC1=NCCc1cccnc1OCCON 81172,N1(C(CCC(=O)Nc2c(CCC)nc(C(=O)OCC)s2)=O)CCc2ccccc21 81173,c1(C(N2CCC(N(C(C3C(OCC)C3)=O)CC)C2)=O)cccc2sccc12 81174,C(=O)(CC(F)(F)C(C)C)NC1CC(CNC(c2c(C)noc2)=O)C1 81175,N1(C(CC2ON=C(CC)C2)=O)CCN(C(c2cnc(C(C)(C)C)o2)=O)C(CC)C1 81176,C1(C#N)(C(=O)NCC2CC(NC(C3(CN(C)C)CC3)=O)C2)CC12CCC2 81177,C1(NC(c2c(OC)n[nH]c2)=O)C2CN(C(=O)Cn3cc(C(=O)NC4CC4)nn3)CC12 81178,N(C(=NCC1CC1)N1CCC(CN2CCOCC2)C1)Cc1c(Br)scc1 81179,C(=O)(C1CCCn2nccc21)NCC1(OC)CN(C(c2c[nH][nH]c2=N)=O)C1 81180,Cc1cc(C(N2CC(NS(=O)(=O)c3nccs3)CC(F)(F)C2)=O)c(Br)cc1F 81181,c1(C(N(c2ncc(SC)cn2)C2CCNCC2F)=O)cc([N+](=O)[O-])c(F)cc1F 81182,C#Cc1c[nH]nc1C(N1CC2CC2(NC(C2CCC(=O)N2)=O)C1)=O 81183,N1(C(c2c(C)n(CC(F)(F)F)nc2)=O)CC2CCCC2(NC(c2cnc[nH]2)=O)C1 81184,c1(CC(N2CC(O)(C3CCCN3C(=O)C=CBr)C2)=O)cccc2ccoc12 81185,CC(CC(=O)NCCCCCNC(C1(O)COC1)=O)c1cccnc1 81186,C#CC1(O)CN(C(=O)C(C)(C)CNC(=O)CC2NC(=O)NC2=O)C1 81187,n1(C(C)C)cnnc1SCC(=O)NC(C)CC(C)NC(c1ccc(C(N)=O)o1)=O 81188,C1(OC)CN(c2cc(NCCCc3ccccc3)ncn2)CCC1F 81189,C1(OCC(N2CC(C(C(=O)NC(C3C=CCS3)CC)OC)C2)=O)CCCOC1 81190,N1(C(CCCNC(C)=O)=O)CC2=C(C1)CN(C(=O)CCOc1cccc(Cl)c1)C2 81191,C1(C(=O)Nc2ccccn2)CC12CCN(Cc1cncnc1)CC2 81192,N1(C(CCc2n(C)ccc2)=O)CCCC2(CNC(=O)CCc3cnc[nH]3)CC12 81193,CC(C)C(C)(CNC(C1C(C)CN1C(C1C2CCC(F)C12)=O)=O)C(C)C 81194,C(=O)(C(C)CCCC(C)=O)NC(CC#C)(C)C(=O)NCC1(O)CC=CC1 81195,N1(CCNC(=O)CC2(F)CN(C(c3cc(CCO)on3)=O)C2)CCNC(=O)C1 81196,C12(C(=O)NC3CN(C(C)C)C(=O)C3)C(NC(=O)CCOCC3CC3)C3CC1C2C3 81197,c1(CC)nc(=N)[nH]cc1C(=O)NC1CCC1NC(=O)CSCc1ccccc1Cl 81198,c1(COC)nc(C(F)F)cc(=NCC2CC2)[nH]1.c12ccc(cc1)NC(=O)C21CC1 81199,N1(C(C(N2CC3C(N)CC(CCC3)C2)=O)=O)CC(F)(F)C2(CCOCC2)C1 81200,C1(CNC(c2scnc2C(F)F)=O)CCCCN(C(=O)CC2CCOCC2)C1 81201,C1(NC(C(C)C2CC2)=O)C2CCC1N(C(c1cccc(-c3nnco3)c1)=O)C2 81202,CC12CN(C(=O)C3=CCC3)CC1(C)CN(C(=O)CCOC(F)F)C2 81203,c1(C(N2CCCCC(NC(=O)C=CCBr)C2)=O)cc(I)ccc1[N+](=O)[O-] 81204,C(=O)(CS(=O)(=O)C1CC1)N1C(CNC(c2cccc3c2CCC3)=O)CCCC1 81205,Cc1nn(CC(=O)NCCCCNC(C2(CNC(N)=O)CCCCC2)=O)c(=O)o1 81206,C(CCF)(C(=O)OC(C)(C)C)NC(CC)CN1CCOCC1 81207,C12(CNC(C3(n4cc(C5(O)CCCC5)nn4)CC3)=O)CCOCC1C2(F)F 81208,N1(C(C(C)CO)=O)CC2(C1)CN(C(c1c[nH]ccc1=O)=O)CC2CO 81209,N1(C(C2C(C)C2)=O)CCCC2(CCN(C(=O)C=CCN(CC(F)(F)F)C)CC2)C1 81210,C1(CC)CCCC(C(N2CCC(OC)C2)C(=O)NCC2CCCO2)C1 81211,CCCC(CCO)N=c1[nH]c(=NCC2CC2C(=O)OCC)[nH]c2c1COCC2 81212,C1(NC(c2cc(=O)cc[nH]2)=O)CC(NC(C2(N3CCCC3)CCC2)=O)C12CCC2 81213,C(CC(O)C(C)(C)C)N(C(c1cc(C#N)cs1)C(=O)NC1COC1)C 81214,C1(NC(CC2(C)CCN(C(=O)C(F)C3CCC3)C2)=O)C(O)C2CCOC12 81215,C1(C)(NC(c2c(CC)n(CC)nn2)=O)CCCN(C(=O)Cc2cncn2C)C1 81216,C1(NC(CC(CCSC)O)=O)CC2CCC(C1)N2C(c1cncc(Cl)c1)=O 81217,c1(C(N2CC3ON=C(COCC)C3C2)=O)ccc2scc(C)c2c1.C1(C)C(=O)N1 81218,c1(C(=O)NC(CN(C(C=CC)=O)C)CC)cc(Br)c2[nH]nnc2c1 81219,N1(C(CC2CCC(C)C2)=O)CC2(CC(NC(=O)CSc3n[nH]c(O)n3)C2)C1 81220,c1(C(=O)NCC2C(OCC)CN(C(=O)C(C)(C)C)C2)cc(C)c(C)cc1N 81221,C1(N(c2nnc(C(N)=O)s2)C)CCCN(C(=O)C(C)(C)CC2CCOCC2)C1 81222,N(C1CC(C)n2ncnc21)C(C=CCNC(c1cccc(C)c1O)=O)=O 81223,N(C1CC2(CCN(C(=O)CC#N)CC2)Oc2ccc(C)cc21)C(C=COCC)=O 81224,N1(C(=O)CC2CC2)CCCC1C1CCCN1C(C1CC1c1ccccc1)=O 81225,N1(C(C2CCCC(=O)O2)=O)CC(NC(C2C3COCC23)=O)C2(CCC2)C1 81226,C(=O)(CC(C)CNC(=O)C=Cc1cncn1C)NC(c1cncnc1)C 81227,N(C1CCSc2ccc(Cl)cc21)C(C1COCCN(C(C2CN(C)C2)=O)C1)=O 81228,Fc1cc(-c2ncc(CN3CCCC(CN4CCOCC4)C3)s2)cc(Br)c1 81229,N1(C(CSCCC=C)=O)CCCN(C(c2cc(F)ncc2OC)=O)C(C)C1 81230,c1(C(N(CCNC(Cn2c(=O)ccc(C)c2)=O)C)=O)cc(F)c(Cl)cc1F 81231,C1(CNC(COCCCC#C)=O)CN(C(C2CC(Cl)(Cl)C2)=O)CCC12CCC2 81232,C1(CCC)(NC(C2CC(=O)N(C)C2)=O)CCN(C(c2cc(F)cc(F)c2)=O)CC1 81233,c1(OC)cc(C)c(Cl)cc1S(=O)(=O)NC1C2CN(C(c3cc(C)on3)=O)CC12 81234,N1(C(c2cnc(C)[nH]c2=N)=O)CC2(CCN(C(=O)CSc3n[nH]c(C)n3)CC2)C1 81235,c1(OC)nc(C)ccc1C(=O)NCCC1CN(C(=O)CC(C)C)CCCO1 81236,N1(C(C(C2CN(C(c3nc(CCC)oc3)=O)C2)OC)=O)CCc2nncn2CC1 81237,C1(C2CCC(=O)NC2)(C(=O)NC2C(NC(C(C)(C)C#N)=O)CCC2)CCC1 81238,c1(C(=O)NC2CN(C(c3c(C)cco3)=O)C(C)(C)C2)c[nH]c2ccccc2c1=N 81239,C(C(=O)NC(C1CCCC1)CO)(C(C)(C)O)NC(c1c(C)nc(C)s1)=O 81240,c1(CC2(C(=O)NC3C(NC(c4c(CC)non4)=O)CC3)CC2)ccccc1Cl 81241,c1(C(=O)NC2CN(C(c3c(CCC)nco3)=O)C2)ccncc1I 81242,[nH]1cc(C(C)(C)C)cn1.C1(NC=O)CCC(CCNC(C2(C3CC3)CCC2)=O)C1 81243,CCCCCC(C(=O)NC1CC2C(NC(C3CC(OC)C3)=O)C2C1)C(C)C 81244,S(=O)(=O)(c1ccccc1Cl)N1CCCC(CNC(c2cnc(Cl)cn2)=O)C1 81245,N1C(NCCC2CCCC2)=NCCCNC2CC12.c1(N(C)C)ccccc1 81246,CCCCCCC(CC)(CC)C(=O)NCC(C)(O)CNC(C1CC(=C2CC2)C1)=O 81247,C1(NC(N2CCC(c3ccccc3)C(F)(F)C2)=O)COc2ccccc2C1 81248,Cc1oc(C(=O)NC2CC2NC(=O)CCc2ccc(C(C)C)cc2)cc1Br 81249,C1(C(=O)OCC)OCCNCC1N(c1ncc(F)s1)C(c1sc(=N)[nH]c1C)=O 81250,N1(C(C#CC(C)(C)C)=O)CCCC12CCN(C(C1(CCF)CC1)=O)CC2 81251,c1(N2CCC(C(=O)NC3CC(C(F)(F)F)C3)C2)ncc2scc(Br)c2n1 81252,N1(C(C(C(C)F)C)=O)CCC(F)(C(F)(F)F)CC1.C12(CCCCC1)C(=O)OCC2 81253,CC1CC(C)CN(C(=O)CN2CCCC(N)C2)C1.C(=O)(CCc1cnoc1)NC(C)C 81254,c1(C(=O)OC)ccc(C(=O)NC2CN(C(=O)Cc3cc(C)no3)C2)cc1C 81255,c1(C(=O)NC2C3CN(C(C(C)OCC)=O)C2C3)ccc2nc(C)n(C)c(=O)c2c1 81256,Cc1c(Cl)cccc1S(=O)(=O)NC1C2CN(Cc3ccc(Br)[nH]3)CC12 81257,c1(NC(C(c2cnc(COC)s2)OC(F)F)=O)cc(Cl)ccc1OCCCF 81258,C1(NC(=O)C(c2ccc(F)cc2)CO)CN(C(c2ccnnc2)=O)CC1C(F)F 81259,CC1(C)CCC(CNC(=O)CC2CCCNC2=O)N(C(=O)C=Cc2cnc[nH]2)C1 81260,c1(C(=O)NCC2CN(C(=O)C(F)Cc3ccccc3)CC2O)cc(O)ncc1F 81261,c1(C(C)(C)C)nnc2n1CC(C(=O)Nc1cc(CC(=O)O)ncn1)CC2 81262,N1(C(COc2cc(C)on2)=O)CC(CO)C2(C1)CN(C(=O)CCC(C)O)C2 81263,C=CC(C)(C)CN=C(NC(C1CC1)C1CC1)NC1CC12CCC2 81264,C(C(C(C)C(C)C)NC(=O)C=CCCC=C(C)C)NC(C1(CCOC)CCC1)=O 81265,C#Cc1cccc(CNC2(c3nnnn3C(C)C)CN(C)CC2C)c1 81266,CCCC(C)(CC)C(=O)NCC1CN(C(c2cnn3c2N(C)CC3)=O)CCO1 81267,CC#CCCCC(=O)N1CCC(CNC(c2noc(-c3ccccc3)c2C)=O)C1 81268,C1(CNC(C(C)Cc2ccncc2)=O)CCCCN1C(=O)COC1CCCOC1 81269,O=C1CCC(CC(=O)NCC2CC(F)(CNC(c3ccco3)=O)C2)CC1 81270,N1(C(CSc2cccc(C)c2)=O)CC2CC(NC(c3ccc(C(C)C)s3)=O)C1C2 81271,c1(C(=O)NCC2C(NC(C3(CN(C)C)CCCC3)=O)C2)cnc(S)nc1 81272,N1(C(COCC#C)=O)CCC2C(CCCN2C(C2Cc3nnc(C)n3C2)=O)C1 81273,C1(C(C)(C)C)(CNC(C2(C)CNC(=O)C2)=O)CCN(C(=O)C(C)(C)c2ccno2)C1 81274,C1(NC(c2cc3ccccc3s2)=O)CC2(CCCCN2C(=O)CCC2CC2)C1 81275,CCC(CNC(=O)Cc1cccn1C)(CC)NC(=O)CCCC#N 81276,N1(C(c2nc(C(C)(C)C)sc2)=O)CCC(NC(C2SCCCS2)=O)C2(CCC2)C1 81277,c1(C(=O)NCC(CNC(C(N2CCOCC2)C)=O)C)n[nH]c2c1COCC2 81278,c1(C(=O)NCC23C(CN(C(C(COC)(C)O)=O)C2)C3)ccc2ncc(C)n2c1 81279,N1(C(C)=O)CCOC(C(=O)NC(C)CCNC(=O)COCc2ccc(C)cc2)C1 81280,c1(C(C2CCCC2C(C)(C)C)C(=O)NCC)cc(C(C)C)ccc1F 81281,Cc1cc(F)c(C(=O)NC2CCOCC2NC(=O)C(C)(C)N(C)C)cc1Br 81282,O=C1CCc2c(C(=O)NCCCCNC(c3cc4ccncc4s3)=O)cccc21 81283,C1(N(C)C(C2CC2C2(C)OCCO2)=O)CCN(C(=O)CSS(C)(=O)=O)CC1 81284,C=CCC(C)(CC)C(=O)N1CCC(CNC(c2ccc(Cl)c(C)c2)=O)C(F)(F)C1 81285,CCC(C)CC(C(=O)N1CC2CC=CC1C2)NC(c1cn(C)nc1OC)=O 81286,c1(OC(C(=O)NS(CCCC)(=O)=O)C)cccc2ccccc12 81287,c1(C(=O)NC)ccc(C(N2CCC(CCCNC(=O)CC(C)(F)F)CC2)=O)cn1 81288,C1(CCC)CN(C(=O)Cc2scnc2C)CCN1C(=O)C(C)SC 81289,c1(C(=O)OC2C(C)CC(=O)CC2)cnc2cc(Br)ccc2c1.C1C(=O)O1 81290,n1(CC(OCC)COC(C)C)c(N2CC3CC3C2)nnc1CNC.C1CCC1 81291,C1(C(=O)N(C)CCc2cnc[nH]2)(NC(C(OC)OC)=O)CCC(C)(C)C1 81292,c1(OC)cscc1C(=O)NC(C)(CNC(=O)CSc1nc[nH]n1)CO 81293,c1(C(N(CC(C)(C)NC(c2c(OC)nsc2)=O)C)=O)c(C)ncc2ccccc12 81294,c1(-n2c(C3CC3Cl)nc(CCOC)n2)ccc(Br)c(F)c1 81295,C1(NC(=O)Cn2nnnc2C2CC2)CCC(NC(=O)C(F)C2CC2)CC1 81296,c1(OC)cc(C(=O)NCC2(OC)CN(C(=O)C(C)CC(N)=O)C2)ccc1C(F)F 81297,C1(CNC(C2C(CC)C2)=O)CC(F)(F)CN1C(=O)CCc1n[nH]c(=N)s1 81298,N1(C(c2ccn(CCN(C)C)n2)=O)CCOC(CNC(C2CC3(CSC3)C2)=O)C1 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81455,Cc1nn(C)c2c(NCc3cnn(C)c3)nc(=NCc3ncc(Br)s3)[nH]c12 81456,c1(CC)cccc(NC(C2CC3CC3N2C(C2CCC(C(=O)O)CC2)=O)=O)n1 81457,C1(CC)(NC(c2nccn2C)=O)CCN(C(C2(c3cccnc3)CC2)=O)CC1 81458,N1(C(C2C(C)OCCN2C(=O)CCN=[N+]=[N-])=O)CCC2(CCCCC2)C1 81459,c1(OC)c(CC(N2CC3(NC(=O)Cc4nc[nH]n4)CCC2C3)=O)cccc1Cl 81460,c1(C(=O)NCC(CNC(c2ncsc2Br)=O)OC)ccc2c[nH]nc2c1 81461,CCC(CC1CCCC1)C(=O)NC(C)CN(C)C(c1c[nH]nc1-c1ccsc1)=O 81462,CC(C)CCC(=O)C(=O)NC1(C(=O)NCC2CCCCN2C)CCSC1 81463,c1(C(N2CCOC(C)(CCOC)C2)C(=O)NC(CC)(C)C)ccc(O)cc1OC 81464,c1(C(N2C(C)CC(NC(CSCC(=O)OC)=O)C2)=O)ccc(OC)c2ccsc12 81465,C(=O)(CCS(C)(=N)=O)N(C(C)CNC(c1csnn1)=O)C 81466,C1(C(=O)NC2(CCCNC(CC3CCN(C)C3)=O)CC2)CN=C2N=CNN2C1 81467,CCC(F)(F)C(C)(C)C(=O)NC1CC(CCNC(c2cn(C3CC3)nn2)=O)C1 81468,C(=O)(CC1CN(C)c2ccccc21)N1CC(COC)(CNC(C2CC2(F)F)=O)C1 81469,c1(C(N(CC(C)NC(=O)C(O)C2CC2)C)=O)sc2cc(F)ccc2c1Cl 81470,CC(C)CC(CNC(=O)CCCOc1ccc(Cl)cc1)NC(C1CC1C(F)F)=O 81471,CCC(C(=O)NCC(C)(C)COC)N(C)C(c1sccc1CO)=O 81472,c1(OC)ccc(-n2cc(C(C)NC(C3CCCC3CF)=O)nn2)cc1OC 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81508,C(C)(c1ccccc1OC(F)F)=CC(=O)NCCC1CC(NC(COC)=O)C1 81509,N1(C(CN(C(c2ccc(C#C)nc2)=O)C2CC2)=O)CC2(CCCN2C)C1 81510,CC1(C)CN(C(=O)Cc2cc(Cl)ccc2Cl)CC1NC(C1(O)CCOCC1)=O 81511,N1(C(CNC=O)=O)CCSCC1C(=O)NCc1cncs1 81512,CC1CN(C(=O)Cc2cc(F)cc(F)c2)CC2(CCN(CCC3CCCC3)C2)O1 81513,C(=O)(C1=CS(=O)CCC1)NCC(C(C)(C)C)NC(COCC(C)(C)C)=O 81514,c1(N(CCCNC(c2cc(C)nc(C)c2)=O)C)cc(C)c(C#N)c(C)n1 81515,CC1(C)CCCC1CNC(c1csc(CNC(c2cscn2)=O)c1)=O 81516,C12(NC(CCOCC)=O)COCCC1CN(C(=O)CNC(=O)CC)C2 81517,C1(NC(c2n(CCOC)nnn2)C2CC=CC2)CC2(C1)CC1CCC2C1 81518,C(C(=O)NNC(=O)Cc1ccccn1)SCc1nnc(C(N)=O)o1 81519,CCC1=NOC(C(=O)N(CCCNC(c2snc(Cl)c2Cl)=O)C(C)C)C1 81520,N1(C(=O)NCC)CCC(Nc2cc(-c3cccc(Br)c3)ncn2)CC1C 81521,C1(CNC(c2c(C)cc(C)o2)=O)CCCCCN1C(C12CC(C(F)F)(CO1)C2)=O 81522,C(C(C)(O)C(=O)NCC1CN(C(c2c(C)noc2C2CC2)=O)CCO1)OC 81523,c1(C(=O)NCC(CNC(CCCOC)=O)(C)F)nccnc1C(N)=O 81524,N1(C(c2cnn3c2OCC(F)C3)=O)CCOc2c(Cl)cc(Br)cc2C1 81525,CCCCCCCC(=O)N(CCN(C(=O)CCC(F)F)CC)CC 81526,N1(C(C(C(CCC)NC(=O)CCCC(C)=O)O)=O)Cc2ccc(O)cc2C1 81527,CC1Cc2ccccc2C1NC(C1(Cc2cc(F)cc(F)c2)CC1)=O 81528,c1(C(C)=O)cc(C(=O)N(CCC(C(C)C)NC(c2cnn(C)n2)=O)C)oc1C 81529,c1(C(N2C(C)(CNC(=O)C=CCF)CCC2)=O)cc2n(n1)CCCC2=O 81530,c1(NCC)cccnc1C(=O)NCC1CN(C(C2CC3C=CC2C3)=O)CC1C 81531,N1(C(Cc2nnc(C)o2)=O)CC(CNC(=O)CCC2CCOC2)C(C)C1 81532,CC1CN2CCN1C(C(=O)NC(C)CN(C(=O)COc1cccc(F)n1)C)C2 81533,N1(C(C2CCC(C)(C)O2)=O)CCN(C(C2CCC(=O)N2)=O)C(C(F)F)C1 81534,C1(N(C(C(C)NC(=O)NC)=O)C)CCCCN(C(=O)C(C)(C)C(=O)OC)C1 81535,Cc1sc(O)nc1C(N1CC(CC(=O)NC(c2cn(C)nn2)C)CC1C)=O 81536,c1(C(N2CCCC(C3N(C(CC)=O)CCC3)C2)=O)ccc2c(C)cc(Cl)nc2c1 81537,C1(NC(=O)C2CC2)CC(O)CN(C(c2ccc(N3CCCS3(=O)=O)cc2)=O)C1 81538,O=C(C1=C(Cl)CCCC1)N1CCCC(CCCCNC(C2(O)CC2)=O)C1 81539,N1(C(C(C=C)CC)=O)CCC(C)C(CC(=O)NCCC2(C)CCOC2)C1 81540,C1(C(N(C2CC(NC(=O)CC3(C)CCOCC3)C2)C)=O)CCC(C(N)=O)N1C 81541,c1(C(N2C(CNC(c3cc(C)cc(O)n3)=O)C(C)CC2)=O)ccn2ccnc2c1 81542,c1(C(N2CC(O)(CNC(C(CC)OC)=O)C2)=O)cc2n(n1)CCCC2=O 81543,c1(C(N2CC(C)(NC(=O)CCC3CCCC(=O)N3)C2)=O)cnc2nccnc2c1 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81944,N1(C(CCCC#C)=O)CCn2c(C(=O)Nc3ccc(Br)cc3C#N)cnc2C1C 81945,C1(OCC=C)CCN(C(c2occc2CNC(=O)CC2(C)CCOCC2)=O)CC1 81946,CC1CCC=C1C(=O)NC(C)C=CC(=O)NCCc1ncc[nH]1 81947,C1(CNC(c2n(CC)ncc2Cl)=O)CCC2(CN(C(C3OCCO3)=O)C2)O1 81948,c1(OC)ccc(C(c2nnnn2C)NCC(c2ccncc2)N(C)C)c(Cl)c1 81949,c1(C(COC(C(N2C(=O)NC3(CCCC3)C2=O)C)=O)=O)ccc(O)c2ccccc12 81950,C(=O)(C1=CCOC1)N(CCC(C)NC(Cc1n(C(C)C)cnn1)=O)C 81951,CCCCCCCC(=O)N1CCC(C)C1CNC(c1ccc(N2CCC2)nc1)=O 81952,C1(NC(CCSCCCC)=O)CC12CCC(NC(=O)C#CC1CC1)CC2 81953,N1(C(C(CC)F)=O)CC2(CC(NC(=O)CCC(C)(C)c3ccccc3)C2)C1 81954,N1(C(c2c(C)cc(O)cc2)=O)CCC(C2CC2)(NC(c2cnc3sccn23)=O)C1 81955,N1(C(c2c(C)n[nH]c2C)=O)CC(NC(=O)Cc2ccc(Br)cc2I)C2(CC2)C1 81956,c1(OC)c(C)csc1C(=O)NC1CC(CCn2cc(C(O)CC(C)C)nn2)C1 81957,n1(CC)ncc2c1CC(C(=O)NC1CN(C(=O)CCc3cncs3)CC1C)CC2 81958,N1(C(C2C(=C)C2C(=O)OC)=O)CC(CNC(=O)Cc2ccc(Cl)cn2)C(F)C1 81959,C1(NC(C(C)=C2CC2)=O)CC(C)(C(=O)NCc2ccnn2C(C)C)C1 81960,c1(OC)cc(Br)cc(F)c1C(=O)Nc1cnn2c1CCCC2 81961,C(=O)(C(O)CCC(C)C)NC(C(C)NC(c1cc(C)c(C(F)(F)F)cc1)=O)(C)C 81962,C1(C(=O)NCC2(O)CCCC2)CC2CCC(C1)N2C(C1CC1C(F)(F)F)=O 81963,N1(C(=O)COc2cccnc2Cl)CCN(C(=O)CCn2cncn2)C(CCO)C1 81964,c1(C(=O)NC(CN(C(c2ccccc2N(C)C)=O)CC)C)ccn(C)c1C 81965,C1(NC(C2C(C)(C(C)C)C2)=O)CCCC2CN(C(C3C=CC=CC=C3)=O)CC12 81966,c1(NC2C(CC)CN(C(C3CCC(=O)N(C)C3)=O)CC2)nccc(S(C)(=O)=O)n1 81967,C1(C(=O)NCC#CCNC(c2cncc(OCCOC)c2)=O)(CC)CCCCC1 81968,C1(C(N(C)CCC2CCC2)=O)C(O)CCN1C(c1ncn(C)n1)=O 81969,C1(C(=O)OCC)CCCN(CC(=O)NCC(C)NC(=O)N(C2CCCCC2)C)C1 81970,C1(OC(CCC)C(=O)NCC)(CO)CCCN(C(=O)C2=COCC2)C1 81971,C1(CNC(c2cc(C)[nH]n2)=O)CC(F)CN1C(c1nc(C(F)(F)F)cs1)=O 81972,CCC(CC)C(=O)NC1CCCC1CNC(c1cn(C(C)(C)C)nc1C)=O 81973,C1(NC(CCNC(C)=O)=O)CC2COCC(C1)N2C(c1cc(C)nc(O)n1)=O 81974,c1(OCCOC)c(C(=O)NCC2N(C(C(=O)NC)=O)CCNC2)cccc1Cl 81975,C1(OC)CCC2(C(N3CC(O)(C(C)NC(=O)C(n4nccc4C)C)C3)=O)CC12 81976,N1(C(c2n(C(C)C)cnc2)=O)CCC2(CCCCC2NC(=O)C(F)CC2CC2)C1 81977,N1(C(CCc2onc(CC)n2)=O)CC2(CCN(C(=O)C(F)CC)C2)C1 81978,C1(C(=O)NC(CC)CNC(=O)Cc2cc(F)ccc2Cl)CNC(=O)CC1(C)C 81979,CC1CN(C(=O)CCC2CC2)CC1CNC(c1cc(-c2cnn(C)c2)no1)=O 81980,C(=O)(CC(C)(C)CC(F)(F)F)NCCOCCN(C(c1cc(C)sc1C)=O)C 81981,C(=O)(C(C)CC(C)C)N1CC(C(C)NC(c2ccc(SCC)nc2)=O)C1 81982,c1(C(=O)NC2CC(CNC(c3c(CN(C)C)ccs3)=O)C2)ccccc1C(F)F 81983,c1(C(N2CCC(N(CCCC)C(=O)CN(C)C(C)C)CC2)=O)cc(C)cc(Cl)c1 81984,CN1CCCC(F)(C(N2CC3CC3(C(=O)C3CC3)C2)=O)C1 81985,CC1(CCO)CN(Cc2cn(-c3ccc(C(OC(=N)O)=O)cc3)nn2)CCO1 81986,c1(NC2CCCC(N(C)C)C2)c(F)cc(Br)c2cccnc12 81987,C1(CNC(c2c(C)nn[nH]2)=O)CCCCN(C(C2CCCC2(F)F)=O)CC1 81988,N1(C(Cc2cn(CC)nc2)=O)CCN(C(c2cc(C)nnc2O)=O)CC(O)C1 81989,N1(CC(=O)NC2(CC)CCN(C(C34CC3COC4(C)C)=O)C2)CCCCCC1=O 81990,c1(OC)ccc(O)cc1C(=O)NC1CN(C(C2CCN(C(C)=O)CC2)=O)CC1C#N 81991,C(=O)(C1CCOc2ccccc21)NCC1N(C(c2cc(N)cc(O)c2)=O)CC=C1 81992,c1(C(N2CC3C(N(C)C(=O)OC(C)(C)C)(C3)C2)=O)cc([N+](=O)[O-])ccc1O 81993,C(CCCCCNC(=O)CC1COC(=O)C1)N(C(=O)CSCc1ccccc1)C 81994,c1(OC)ccc(C(=O)N(C)C(C2CCOCC2)C)c(C(F)F)c1 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82012,c1(NC(C)=O)c(Sc2nc(N(C(=O)C#CC3CC3)C)sc2)ccc2c1CCC2 82013,c1(OCC(C)(C)C)cccc(C=Cc2nc(CN3CCCOC3=O)no2)c1OC 82014,c1(C(=O)NC2(C(N(CCC(C)C)CC(C)C)=O)CC2C)cccn(C)c1=O 82015,C(=O)(C(C)(C)CCSC)NCC1(OC)CN(C(C2(F)CCCN(C)C2)=O)C1 82016,C1(NC(C(C)N(CC(F)(F)F)C)=O)CC(C)CN(C(c2cc(Cl)c[nH]2)=O)C1 82017,c1(C(N2CC(CC)C(NC(=O)C3=CCOCC3)C2)=O)cnc2ccccn2c1=O 82018,C1(C(=O)NC2(C)CCCO2)COC2(C1)CN(C(=O)CN1CCOCC1)C2 82019,c1(OC)ccc(C(N2CCC(NC(=O)C=Cc3ccn(C)c3)CC2C)=O)cc1F 82020,C1(NC(CCCOCC)=O)COCCN(C(=O)C=CCNC(=O)OC(C)(C)C)C1 82021,c1(COC)cccc(C(=O)NCC#CCNC(=O)CSc2ccccn2)c1 82022,c1(C(=O)NCC2C(NC(C=C(CC)C)=O)CC2)cnn(CCCC)c1C 82023,c1(C(N2CCCC(C)(NC(=O)C=CC3CCOCC3)C2)=O)cnc2sccc2c1 82024,C1(NC(C2(c3cc(C)no3)CC2)=O)CCC(C)N(C(=O)C(C(C)C)C2CCC2)C1 82025,CC(C(C)C(=O)N1CC(C)(F)C1)NC(c1ccc[nH]1)=O 82026,C(c1cncnc1O)=CC(=O)N(C1CCCC(NC(c2n[nH]c(C)c2Cl)=O)C1)C 82027,c1(C(C)NCCOCCN(C)C)cc(F)c(Br)cc1F 82028,N#CCCCCCC(=O)N1CCN(C(=O)C=CC=C(Cl)Cl)C(CO)C1 82029,CC(C)(C(=O)N1CCC(O)(CCNC(C23CC(CCO2)C3)=O)CC1)C(N)=O 82030,CCC(C)(CCC(C)C)C(=O)N1CCCC(CNC(=O)C(C)(C)COCC)CC1 82031,N1(C(c2ccc(C(C)(C)C)[nH]2)=O)CCOC2(CCC(NC(C3CCO3)=O)CC2)C1 82032,C1(NC(c2c(C)sc(O)n2)=O)CN(C(c2cc(F)cnc2O)=O)CCC1C 82033,C#Cc1cccc(C(=O)NCCC(C)(C)NC(=O)COCc2ccccc2)c1C 82034,c1(CN(C(=O)CC=CCNC(C2CC2C(=O)N(C)C)=O)CC)cncn1C 82035,N1(CC(C)(C)NC(C2N(CC)CCC2)=O)CCN(C(=O)Cc2scnc2C)CC1 82036,c1(C(c2nnnn2C)NC(Cc2c(C)noc2C)C)ccc(Cl)cc1F 82037,CC(F)(C(=O)N(CCNC(C1CCCOC1)=O)C1CC1)c1ccon1 82038,C(=O)(C(C(C)O)N(C)C)NCC1N(C(Cc2ccc(C(C)=O)s2)=O)CC=C1 82039,Cc1nnc2n1CCN(C(C1CC(C)N1C(=O)Cc1nccn1C)=O)C2 82040,S(=O)(=O)(C1CC1)NCC(=O)NCCOCCNC(C1C=CCC1)=O 82041,C1(CCC)CN(C(C2CCS(=O)(=O)C2)=O)CCN1C(c1cccnc1S)=O 82042,N1(C(C2(COC)CC=CCC2)=O)CCC2(CCCCN(C(=O)CC(F)(F)Cl)C2)C1 82043,C(C(C)C(F)C(=O)NC(C)(C)C(O)C(F)F)NC(C1C(=C)C1C(=O)OC)=O 82044,Cc1noc(C)c1C(C)C(=O)NCC(CNC(=O)Cc1cccnc1)CO 82045,c1(CC)nn(C)c(C(=O)NCCN(C(=O)C(CC)C(C)O)C2CC2)c1Cl 82046,C=CC(C)(C)C(=O)NCC12CC(CN1C(=O)C(C)NS(=O)(=O)CCCC)C2 82047,c1(C(=O)NCC2CN(C(C=C3CCN(C)C3)=O)C(C)(C)C2)csc(S(C)(=O)=O)c1 82048,C(=O)(CC1=CCCCC1)NC1C(C(N2CC(C(C)C)OCC2)=O)OCC1 82049,C1(NC(=O)C2CC2)CC2CCC1CC2NC(C1CCC(c2ccccc2)CC1)=O 82050,S(=O)(=O)(CC(=O)NCCC1CN(C(=O)Cc2cc[nH]n2)C1)NC(C)(C)C 82051,C1(C)(CNC(COC2CN(C(C)=O)C2)=O)CC1(Cl)Cl 82052,N1(C(Cc2n(C)cnc2)=O)CCOCC(CNC(C2(C3CCCO3)CCC2)=O)C1 82053,Cc1noc(Cl)c1CC(=O)NCC(C)(C)CNC(c1c(C)nsc1N)=O 82054,c1(N2CC(CCOC)OCC2)ncc(C)cc1S(=O)(=O)NC1C=CCC1 82055,Cc1oc(-c2ccco2)nc1CC(=O)NCC(C)(C)NC(=O)CNC=O 82056,c1(-n2c(COc3ccccc3)nc(COC)n2)ccc(F)cc1C(=O)O 82057,c1(C(N(CCNC(c2ccnc(CO)c2)=O)CC2CC2)=O)cccc(O)n1 82058,c1(C(N2CC(C)C(NC(=O)C(c3ccc(F)cc3)(C)F)C2)=O)cccc(Cl)c1N 82059,C1(NC(CCC2(C)CN(C(COCC(=O)NC)=O)C2)=O)CCCCCC1C 82060,c1(C(N2CCC(N(C(CCC(C)C)=O)CCO)C2)=O)ccc([N+](=O)[O-])cc1 82061,N1(C(c2cc(C)[nH]c2)=O)CC2CCC(C(=O)NCC3=NOC4CCCC34)(C2)C1 82062,CCCC(C(=O)NC(C(=O)NC1CCCCC1N(C)C)C1CCCC1)OC 82063,C1(C(=O)NCCCC(C)NC(c2scc(C)c2Cl)=O)CCC(=O)C(C)C1 82064,N1(C(c2cc(Br)n3c2CCC3)=O)CCCC2C1CCCN2C(=O)CO 82065,c1(C(N2CCC(N(C(=O)CC34CCCC3C4)CC)C2)=O)ccc(Cl)c(N)c1 82066,C1(CNC(c2c[nH]nc2C(F)F)=O)CCCCN1C(C1(C(F)F)CC1)=O 82067,c1(C(=O)NC2(C#N)CCN(C(c3cc(O)no3)=O)C2)cccc2ncsc12 82068,C1(CNC(C(C)=C(CC)C)=O)(OC)CCN(C(C2CC(=O)N(CC(C)C)C2)=O)C1 82069,C1(NC(=O)Cn2nnc(-c3ccco3)n2)CCN(C(=O)Cc2cnc[nH]2)CC1O 82070,C=CCC(CC(=O)N1CCC(C)(CO)C1)NC(=O)CCC(C)OCC 82071,c1(OC2(C(N(CCCCN(C(=O)CCC3CC3)C)C)=O)CC2)cnn(C)c1 82072,Cc1cccc(C(O)C(=O)N2CC(NC(=O)C(C(C)C)N3CCCC3)C2)c1 82073,CON(C)C(=O)CNC(c1c(CNC(=O)CC(C)=C(C)C)cnn1C)=O 82074,N1(C(CCC=C(C)C)=O)C2CCC1CC(NC(=O)C(C)N(C)C)C2 82075,Fc1ccc(CNc2cc(NCC(F)F)ncn2)cc1OCC(F)F 82076,Cc1ccc(=NCCC(=O)NCC(C)NC(c2cc3n(n2)CCN(C)C3)=O)[nH]c1 82077,n1(CC)ccc(C(=O)NCCCN(C(=O)C=C(C)C(F)F)C(C)C)c1C 82078,c1(C2C(C(=O)NC(CN(C)Cc3ccc(C)o3)C)C2)ccccc1C 82079,C(C(=O)NCC(O)CC(=O)NCC(Cl)=CCl)(C(C)(C)C)N(C)C 82080,C(=O)(CCCC(C)CC)NCC1CN(C(c2c(C)cc(CC)o2)=O)CC12CC2 82081,C(CC(C)C(=O)NCC1CN(C(C2(CO)CC(C)(C)C2)=O)C1)=CC 82082,Nc1c(F)cc(-c2ccc(-c3nccn3C3C4CNCC34)c(F)c2)cc1F 82083,N1(C(C2C(OC)CCC2)=O)CCC2CC2(C(=O)Nc2cc(O)ccc2F)CC1 82084,C1(N(C(CCCOCC)=O)C)CCN(C(=O)CCSc2ccccc2Cl)CC1C 82085,C1(C(N(CC(C)NC(C2C(C)OCCC2)=O)C)=O)CCCC2C1C2(F)F 82086,O(NC(=O)C(C1(O)CCCCC1)NC(=O)CCC(C)C)C(C=C)C 82087,c1(OC)ccc(F)c(C(=O)NCCC2CCCCN2C(c2csnn2)=O)c1Cl 82088,C1(CC(=O)NCC2CN(C(CCSCCC)=O)C2)CCCNC(=O)C1 82089,c1(C(N2CC(N(C(Cc3ccc(C)o3)=O)C)C2)=O)cccnc1N(C)C 82090,n1(CC)c(C)cc(C(N2CCCC(CO)(CNC(=O)C(O)CC(C)C)C2)=O)c1C 82091,c1(C(N(CC(CN(C(C(CCC)F)=O)C)O)C)=O)cccc(CC)c1F 82092,C12(CNC(c3cc(CCC)nc(O)c3)=O)CCC(CC1)N(C(=O)C(F)=C(C)C)C2 82093,C1(CC(N2CC(COC)(NC(=O)C=CCO)C2)=O)CCOCC1(C)C 82094,N1(C(c2cc(CC)n(CCO)n2)=O)CCN(C(c2ccsc2Cl)=O)C(CC)C1 82095,Cc1cccc2c1ccn2CC(=O)N(C1CN(C(=O)C(F)C(F)(F)F)CC1O)C 82096,N1(C(=O)C=C2CCC2)CCN(C(C2C3CNC(=O)C23)=O)C(c2ccccn2)C1 82097,Cc1c(C(=O)NC2CCC2CNC(=O)CCS(C)(=O)=O)sc2cncn12 82098,c1(OC)ccnc(C(=O)NC(C)CCNC(=O)C=Cc2ccnn2C)c1N 82099,CCC(CCC(=O)NC1CC(OC)CN(C(c2ccc(F)c(OC)c2)=O)C1)OC 82100,c1(C(=O)NCC(CNC(c2cc(C)cs2)=O)OC)cc(O)n(C)n1 82101,N1(C(c2c(COC)cccc2)=O)CCN(Cc2cc(C)sc2C)C2CC12 82102,N1(Cc2c(COC)cncc2)CC(F)(F)CC1COC(c1cccc(Br)c1C)=O 82103,CC1CCC(C)(C=CC(=O)NC2CC3(CCN(C(C4(C)CC4)=O)C3)C2)C1(C)C 82104,c1(C(=O)NC)cc(Cl)ccc1NCc1ccc(C(C)(C)C)cc1.C1(C)C(=O)N1 82105,c1(C(N(CC(C)NC(c2cnc(C#N)s2)=O)C)=O)cccc(N(C)C)c1 82106,c1(CN(c2c(F)cnc(OCC)n2)C2CNCC2O)ccc(F)c(Cl)c1F 82107,c1(CCC(=O)NC23CCN(C(c4ccoc4)=O)CCC2C3)cnc2ncccn12 82108,C1(CNC(c2n(C=C)ncc2)=O)CN(C(C2(C#N)CC3(CC3)C2)=O)CCN1C 82109,C(CCCCCC(=O)NC1CCCSC1)NC(c1ccc(Cl)cn1)=O 82110,c1(CNC(C(C2CCOC2)NC(C(F)=CCC)=O)=O)ncnn1C 82111,C12(NC(CC)=O)CCC(C(N3CCNC(=O)C3C(C)C)=O)(CC1)C2 82112,C(=O)(CC(O)C1CCCC1)N1C(CNC(=O)Cc2csc(Br)c2)CC1 82113,c1(C(=O)NCC2N(C(c3c(CC)ccc(C)c3)=O)CCC2)nc[nH]c2ncnc1-2 82114,N1(C(=O)NC(c2ccccc2)=O)CCN(Cc2occc2Cl)C2CC12 82115,C1(CC(=O)N(C)CC2CN(C(=O)C(C)(C)n3cccn3)C2)(OC)CCCCC1 82116,N(C(=NCCC(C)(O)C1CC1)NC1CCC(N(C)C)CC1)C(CC)C 82117,N1(CCCc2nc(C)sc2)CCCC(CNC(=O)COC2CCCC2)C1 82118,CC(C)(C)CCCC(=O)NC1(C)CCN(C(C2(C)CCCO2)=O)C1 82119,N1(C(C(OC)OC)=O)CC(=O)NCC1C(=O)NCCOCCCF 82120,c1(C(N2CC3CN(C(C(CCC)O)=O)CC32)=O)ccc2cnn(C)c2c1 82121,c1(C(=O)NC2COCCC2NC(C2CCCCO2)=O)ccc2c(c1O)CCC2 82122,C1(NC(c2cnc(CC)o2)=O)CC(NC(c2nc(C)c(C)s2)=O)C12CCC2 82123,C(=O)(C1CCCc2nn[nH]c21)N(C)CC1CCN(C(CCNC(=O)NC)=O)C1 82124,N1(C(CCSC)=O)CC2C(CNC(=O)Cc3scnc3C)C2C1 82125,Cc1c(F)ccc(C(N2CCOC(CNC(C3(C)C=CCC3)=O)C2)=O)c1Cl 82126,CCC(CC)CCC(=O)NC1CCOC(C(N2CCN(CC)CC2)=O)C1 82127,N1(C(CCCCCCC)=O)CCN(C(=O)CCC(C)(C)OC)C2(CCC2)C1 82128,c1(N(C)C)ccc(C(=O)NC2CCC2NC(c2ccncc2F)=O)cc1[N+](=O)[O-] 82129,O=C(NNc1nc[nH]n1)c1ccc2n[nH]cc2n1 82130,C1(NC(c2cnc(CC(C)C)[nH]2)=O)CCSC12CN(C(=O)CCc1nc[nH]n1)C2 82131,C1(C(N2CCCC(OC)C2)=O)COCCN(C2CCCC(C)C2)C1 82132,c1(C(C)(C)C)ccc(CCCC(=O)NC2CCN(C(C3CC34CCC4)=O)C2)cc1 82133,c1(N2CC3C(NC(C(CC)CCOC)=O)C3C2)c(Br)cccc1[N+](=O)[O-] 82134,C1(CC)CCC(O)(C(=O)NCCN(C(=O)CS(C)(=O)=O)C2CC2)C1 82135,n1(CCCO)nc(-c2ccc(OCc3ccccc3)cc2)nc1-c1ccon1 82136,C(N=c1[nH]c(C)ncc1F)C1C(NC(C=CCC)=O)C2(CC1)CCC2 82137,N1(C(c2[nH]c(=NC)sc2)=O)CCCC2(CCC(NC(c3ccc(C)o3)=O)C2)C1 82138,C1(C(=O)NC2CC(C(=O)NC(C(C)C)C)C2)(CF)CCOCC1 82139,Cc1cc(N)ccc1C(N1CCC(O)(CCNC(c2ccnc(CO)c2)=O)C1)=O 82140,c1(C(N2CCCC(Nc3cc(C)nc(C)n3)C2)=O)cc(C)c(F)cc1F 82141,C1(C(N2CC(CNC(=O)Cn3cncn3)C2)=O)CC(O)CN1c1ccncn1 82142,N1(C(C2CCC(CNC(CC(C)F)=O)C2)=O)CCOC2(CCCC2)C1 82143,C1(CCNC(N2CC(c3ccc(Cl)nc3)C2)=O)CCC2(CCC2)O1 82144,C(=O)(CCCCC(C)(C)C)NCC(COC)NC(=O)CCc1csc(C)n1 82145,c1(C(N2CC(NC(=O)OC(C)(C)C)CC2C)C(=O)NCCSC)nc(C)n(C)n1 82146,N1(C(COC(CC)(C)C)=O)C(CNC(c2ccc(C)nn2)=O)CC2COCC12 82147,N1(C(c2cc(OC)no2)=O)CCCCC1C1(NC(=O)CCc2cncnc2)CC1 82148,N1(C(C(C)CF)=O)CCOC2CCN(C(c3ccc(N(C)C)cc3)=O)CC12 82149,CC(CC(F)F)C(=O)NCC1CCCCN1C(=O)CCCNC(N)=O 82150,N1(C(CCc2scc(C)c2)=O)CCN(C(N2CC(c3ccccc3)C2)=O)C(=O)C1 82151,c1(OC)cc(F)c(S(N)(=O)=O)cc1C(N1CCC(N2CC(F)C2)C1)=O 82152,n1(CCOC)cccc(C(N2CCOC(C3CCCCC3)C2)=O)c1=O 82153,C1(CC#C)CCN(C(C2CCC(NC(=O)CCC3CC3C)CC2)=O)CC1 82154,C1(C(=O)NC2(CF)CN(C(C3C(C)CCC3)=O)C2)COCCN1C=O 82155,N1(C(C2CCN(Cc3ccc(C#N)s3)CC2)=O)CC2CCC(C1)O2 82156,c1(NC(C2CCN(C(c3cccc(C4(C)CC4)c3)=O)C2)=O)ncc(Br)cc1C#N 82157,C12(C(=O)NC3(C)CC(NC(C(C)Cc4ccncc4)=O)C3)CCC(C1)OC2 82158,N1(C(C2(CCC=C)CN(C(C3C4C5CCC(C5)C34)=O)C2)=O)CC(O)C(C)(C)C1 82159,c1(OCC)ccc(CC(=O)NCCC2CN(C(C3CN(C)C3)=O)CC2C)nc1 82160,c1(C(=O)NCC(c2ccccc2)NC(=O)CCC2CC2)cnn2c1OCC(O)C2 82161,C1(C(=O)NCC(CNC(=O)CCc2ccc(Cl)cc2)F)NC(=O)C2CCC12 82162,N1(C(c2cnc(OC)nc2)=O)CC2CC(NC3CN(C(=O)OC(C)(C)C)C3)C2C1 82163,c1(C(C(=O)NC(C)C(CO)NC(c2ccc(CO)o2)=O)O)ccc(F)cc1 82164,c1(N2CC(O)(CCNC(C3CCC(C)C3)=O)C2)cc(F)ncn1 82165,C1(C(=O)NCCC(CCC)O)C2CCC(C2)N1C(c1coc(N(C)C)n1)=O 82166,C(=O)(CCCCCN(C(=O)C(F)C(C)(C)O)C)N(CCC#C)CCO 82167,N1(C(COC(C)C)=O)CCC(O)(C(C)NC(=O)CCc2cnn(C)n2)C1 82168,Cn1cc(C(=O)NCCCC2CCN(C(c3cccc(CF)c3)=O)CC2)nc1O 82169,C1(OC(c2cncc(OC(C)(C)C)n2)=O)CCC=CCCC1 82170,C(c1cccc(Cl)c1)=CC(N1CC(NC(c2ccc(OCC)nc2)=O)C(O)C1)=O 82171,C1(NC(C2CCCC3(CCC3)C2)=O)CN(C(C2CC(F)(F)C2)=O)C2CCCCC12 82172,N1(C(c2ccc(OC)nc2)=O)CC(NC(=O)Cn2nnc(=O)[nH]2)CC12CCOC2 82173,c1(CC(=O)NC2CCCC(CNC(COCCC(C)C)=O)C2)ccc(C#N)nc1 82174,CC1CCOCC1C(=O)NCC1(C(=O)NC2CC(=O)N(O)C2)CCCCC1 82175,c1(C(N(C2C(N(C(=O)CCF)C)CCCC2)C)=O)cnn2c1CCCC2 82176,O=S(=O)(c1ccc(Br)cc1NCCCCCCSC)NCC1(c2ccon2)CC1 82177,c1(C(C)NC(C)CC2CCCC2)ccc2c(c1)CCCC2 82178,C1(CC(=O)NC(Cc2cn[nH]c2)C(=O)NCCN2CCOC2=O)CCCNC1=O 82179,C1(C(=O)NCC(CNC(c2ccc(C(=O)OC)cn2)=O)O)C(F)(F)C12CCC2 82180,c1(SCCOC(C(COC)(C)OC)=O)nnc(O)c2ccccc12 82181,C1(C(N2CC(COC)(CNC(c3cocn3)=O)C2)=O)CC2(CSC2)C1 82182,c1(CCC)cccc(NC(=O)CCC2CC(NC(=O)C(C)SC)C2)c1 82183,c1(C(=O)NCc2ccc(CNC(C3C(C)CCO3)=O)cc2)ccc2nn[nH]c2n1 82184,N1(C(c2c(C)cc(C(F)F)o2)=O)CC(C)N(C(C2CCNC(=O)C2)=O)C(C)C1 82185,C(N=c1cccc(S(=O)(=O)NC2CCCc3occc32)[nH]1)c1c(C#N)cccc1 82186,c1(-c2ccn(C)n2)cc(C(=O)Nc2cc(Cl)nc(Cl)c2)cc2cc[nH]c12 82187,Cc1cc(C(=O)NCc2n[nH]cc2C(=O)N(C)Cc2cnn(C)c2C)c(C)nn1 82188,N1(C(c2c(OC)cc(Br)c(C)c2)=O)CCC2(CCCC2C(=O)N(C)C)C1 82189,N1(C(c2c(C)snc2)=O)CC2CC3CC2C1C3NC(=O)CC1OCCC1C 82190,c1(NC2C(C(=O)OCC)CNCC2)ccc(-n2cccc2)c(Cl)c1 82191,c1(OC)nc(C)c(COC(=O)CCC2CC(C)(C)CO2)s1 82192,C(=O)(CCC(=O)NCC1(C(=O)NCc2ccn(C)n2)CC1)NCCC 82193,c1(NC(C)=O)cc(C)c(Br)cc1C(=O)NC(C)C(c1ccccc1F)O 82194,c1(NC(C2C(C(=O)Nc3cc(C(C)(C)C)[nH]c3)C2)=O)c(O)cccc1Cl 82195,c1(C(=O)NC(C(=O)NC2(CO)CC(C)C2)c2cccs2)cc(C#N)cs1 82196,CC(CC1CCC1)N=c1[nH]c(=NC2CCn3c(O)nnc3C2)[nH]c2c1COCC2 82197,c1(C(C(N2CC(CC)C(NC(=O)C(C)NC(C)=O)C2)=O)(F)F)ccc(F)cc1F 82198,N1(C(C2CC(OC)C2)=O)CC2(CCN(C(C3CCC=CCCC3)=O)C2)C1 82199,Cc1ccc2nc(C(N3CCN(C(=O)CC4(CO)CC4)C(CO)C3)=O)cn2c1 82200,C1(CNC(Cc2ccc(SCC)cc2)=O)CCCCN(C(C2OCCCO2)=O)C1 82201,C1(CNC(c2c(C)cnn2C(C)C)=O)CN(C(=O)CCCC2CC2C)CC1(F)F 82202,c1(C(=O)NC(CN(C(C2CCC(C)O2)=O)CC)C)ccc(N)c(C(F)(F)F)c1 82203,C1(=CC(=O)N(C2CCC(NC(C(C(C)C)O)=O)C2)C)CN2CCC1CC2 82204,C1(C)(NC(CN(C)C)=O)CCC(NC(=O)CCC2CC(C)(C)CO2)CC1 82205,COn1cnc(C)c1C(=O)NCc1nc(C)c(C(=O)NCC2C=CCC2)o1 82206,CC1(NC(=O)Cc2csc(S)n2)CCCN(C(C2CCCC2(F)F)=O)C1 82207,N1(C(C(C)OCCOC)=O)CC(CNC(=O)C(N2CCC(C)CC2)=O)C(O)C1 82208,C(c1cnn(C)c1)=CC(=O)NCC(CCNC(=O)C(C)(C1CC1)OC)OC 82209,C(CNC(=O)Cc1cccs1)(CC(=O)NCCC1CC(F)C1)OC 82210,n1(C(C(=O)NC(C)CSC(F)F)C)cc(C2(N3CCC3)CCC2)nn1 82211,C1(OC)CC2CCC1CC2C(=O)NC1CN(C(=O)C(C)Cc2ccc(C)cc2)C1 82212,c1(CCNC(CC2(C(=O)OC)CC2)=O)cccc(OCC=C(C)C)c1 82213,c1(C(N2CC3CCN(C(C4CC(C)(O)C4)=O)CC32)=O)cnc2ccc(F)cc2c1 82214,C1(CNC(C2(OC)CCCCC2)=O)CC2CN(C(C3CCN(OC)CC3)=O)CC12 82215,c1(CN(C(=O)Cn2ccnc2C)CCNC(C(COC)O)=O)ccc(F)cc1 82216,C12(CNC(c3c(OC)nn(C)c3)=O)CCC(CC1NC(=O)CC1CC(F)(F)C1)C2 82217,c1(OC)cc(Cl)c(N=c2nc(Oc3ccco3)[nH]c(C(N)=O)n2)cc1Cl 82218,C(=O)(C(C(C)NC(=O)C=Cc1cc[nH]n1)C(C)C)NCCC 82219,c1(C(N2C(CC(=O)NCCCc3cc[nH]n3)COCC2)=O)occ2c1CCC2 82220,C1(CNC(CN(C)C2CC2)=O)CN(C(=O)CC2NC(=O)NC2=O)CCC1(C)C 82221,C1(C(NOCC(C)(C)O)=O)C2CC3C(C2NC(C2CCCC(=O)CC2)=O)C13 82222,Cn1cc(C(N2CCN(C(=O)COC3(C)CCCC3)C(C3CC3)C2)=O)ccc1=O 82223,C1(C(N(C2CC(=C)C2)C)=O)C=CCCN1C(=O)C(C)OCOC 82224,C1(CC(N2C(CCN(C)C(C3CCCS3)=O)CCCC2)=O)CCC2(CC1)CC2 82225,c1(CC)nc(N2CCC(NC(=O)CSCCN(C)C)C(F)C2)c(C)c(Cl)n1 82226,Cc1sncc1C(=O)NCC(C)C(=O)NCCNS(N)(=O)=O 82227,c1(C(=O)NC(C2CN(C(=O)COC(C)(C)C)CCO2)C)noc2ccc(F)cc12 82228,C1(C)(C(N(C2CCCN(C(C3(C#N)CCCC3)=O)CC2)C)=O)CCC(=O)NC1 82229,N1(C(C2(CC=C)CCCN2C(=O)C2=CCOCC2)=O)CCC2OCCC2C1 82230,c1(C(N2CCCC(CNC(CC(C)SC)=O)C2)=O)nn(C)c(Cl)c1Cl 82231,C(C1CCCN1C(=O)C(C)n1ccnn1)=CC(=O)NC1(C(COC)O)CC1 82232,CN=c1[nH]cc(C(N2CCC(OCCNC(c3cc(C(N)=O)co3)=O)C2)=O)s1 82233,C1(CC(=O)NC(CNC(CCOC(C)C)=O)CO)CCOC1(C)C 82234,C(CC(=O)N1CC(C)(NC(C2CC3(C2)CS(=O)(=O)C3)=O)C1)(C1=CCCC1)OCC 82235,C(C(CN=c1[nH]c(=NC2CC3CCC(C2)O3)[nH]c2c1CSC2)OC)OC 82236,C12(C(=O)NCCOCCCC)CCC(CC1NC(=O)C(C)CCOC)C2 82237,C1(O)CC1.C1(=O)C=CC(=O)N(C)CC2(CC2)CN1.C(=O)(CNC=O)N(C)C 82238,C1(CC)CN(C(=O)Cn2cccn2)CC1C(=O)NCC1CCCOC1 82239,C(N=c1nc2c(cnn2C)c(N(C)Cc2cc(C)no2)[nH]1)C1(OC)CCCSC1 82240,C1(CNC(CCSCCC)=O)CN(C(c2c[nH]ccc2=O)=O)CC(C)(C)C1 82241,N1(C(CCCN(C(=O)OCC)C)=O)CC=CC(NC(C2C=CCC2)=O)C1 82242,c1(CC(=O)NCC2CN(C(c3csnc3Cl)=O)CC2O)nsc2ccccc12 82243,CC(C)C(C(=O)NCCCNC(=O)Cc1cccn1C)c1cccc(Cl)c1 82244,C1(C(NOCCCC#C)=O)CCN(C(=O)CSc2ccc(C)cc2)C1C1CC1 82245,C12(CC)CN(C(c3ccnn3CC(F)F)=O)C(CNC(C3CC(C)=NO3)=O)(C1)C2 82246,N12CC(C(C)(C)C1)N(C(C)(C)C)C(=O)CCSCC2=O.Cn1cc(C(=O)C=O)cn1 82247,N1(C(c2c(SC)cnn2C)=O)CC2(CCN2C(c2ccc(Cl)c(C)c2)=O)C1 82248,c1(C(N2C(CNC(=O)CCc3ccon3)CCCC2)=O)ccc2c(c1)B(O)OC2 82249,C(=O)(CCCCCNC(=O)CC1C=NNC1=O)NCCCS(C)(=O)=O 82250,CC1C(C(N2CCC(C(CO)NC(C3CCS3(=O)=O)=O)CC2)=O)CCN1C 82251,c1(CC)conc1C(C(=O)NCC1CC1)N(CCOC)Cc1nnn(C)n1 82252,S(=O)(=O)(c1ccc(I)c(C(=O)O)c1)NC(c1ncccn1)CC 82253,c1(C(C)=O)cn(C)nc1C(=O)NCC(C)(C)CN(C)C(C1C=CCC1)=O 82254,C1(CCOC)(NC(c2ccc(CC(C)C)s2)=O)CCN(C(=O)C=C(C)Cl)C1 82255,CC1C(C)N(C(C2CCn3nccc3C2)=O)CCN1C(C12CC(F)(C1)C2)=O 82256,c1(N(C)C)cccc(C(=O)NC2CCN(C(=O)Cc3csc(Cl)c3)C2C2CC2)n1 82257,N1(C(CCC=C)=O)CC(N=c2[nH]c(Cl)nc(C)c2[N+](=O)[O-])C(C)(C)C1 82258,c1(-c2ccc(C3(SC)CC3)cc2)cnc(C(=O)NC(C)CCCC(C)C)cc1C 82259,c1(C(=O)NC(CCNC(C(C(=O)OCC)(C)F)=O)C)cc2cnccc2o1 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82329,CC1(C)COCC(NC(C2CCC(C)(F)CC2)=O)CN1 82330,C=CC(C)(O)C(=O)N1CC(CNC(c2ccc(OC)s2)=O)C1 82331,c1(C(C)(C)C)ncc(C(=O)NC2CCN(C(=O)CCN3CCCC3=O)C2)s1 82332,Cc1cc(Br)cc(C)c1CNC1CC(C(=O)Nc2nnco2)C1 82333,CC(C)(C#N)CC(=O)NCC1(CCNC(c2ocnc2-c2ccccc2)=O)CC1 82334,C1(N2CCC(NC(c3cnsc3)=O)C2)CCN(C(=O)COC(F)(F)F)CC1 82335,N1(C(C(C)N(C(C)=O)C)=O)CCCCC1CCNC(c1occc1C)=O 82336,C(=O)(C(C(C)C)N1CCCC1=O)N1CCC(CNC(c2n(CC)ccn2)=O)C1 82337,C1(CC(=O)N(CCC(C)NC(c2c(C)noc2)=O)C)CC(=O)NC1=O 82338,c1(CC(N2C(C(=O)NCC(CC)n3cccn3)CC2C)=O)ccc(F)c(C)c1.C(C)(=O)O 82339,c1(NC(N(C)CCN(C2CCOC(c3ccccn3)C2)C)=O)ccc(Cl)c(Cl)c1 82340,C(C(=O)N(CCC(=O)NC1CC(C(C)O)C1)CCO)(C1CCC1)OC 82341,C1(C(N(C2CCCCC2)CC)=O)CCCCC1CNc1sccc1C 82342,n1(CC)nc(C)c([N+](=O)[O-])c1N1CCCC(NC(c2sccc2COC)=O)C1 82343,N1(C(C(C)NC(N)=O)=O)CCC(F)(CNC(=O)CCc2cncnc2O)C1 82344,C(=O)(CC(C)C(=O)NCC(C1CCN(C(C2CCCCCC2)=O)CC1)(C)C)OC 82345,c1(C(N2CCC(F)(C(=O)NC(C3CCOCC3)C#C)C2)=O)ccc(C#N)cc1 82346,C(C(F)(F)C(=O)N1CC(O)(CNC(c2ocnc2C)=O)C1)OC 82347,c1(C(=O)NCC(CCOC)NC(=O)C2=CCCCC2C)cc(C)ccc1[N+](=O)[O-] 82348,CC1=CCC(C)(C(=O)NC2CN(C(c3ccc(CF)cc3)=O)CC2O)CC1 82349,N1(C(c2cc(C)c(C)nc2)=O)CC(NC(=O)CNC(N)=O)C(S(C)(=O)=O)C1 82350,CC(F)(F)C(C)(C)C(=O)N1C2CCC(C(=O)NCC34CC(CCO3)C4)C1CC2 82351,CS(=O)(=O)C1CC2CCC(C1)N2N1CC2CC1(CO)CO2 82352,Cc1ccc(F)c(C(=O)N(C)CC2CCCN(C(C3CCC(C)O3)=O)C2)c1F 82353,Cc1cc(-c2ccccc2)ccc1CNC(CCO)C(C)(C)C 82354,c1(C(=O)NC2CCC(Cn3cc(CS(CC)(=O)=O)nn3)C2)cc2c(s1)CCCC2 82355,Cc1c(C(N2CCC(O)(CNC(c3cncnc3)=O)C2)=O)cnn1C1CCC1 82356,C1(NC(C(C)Cc2cccc(Cl)c2)=O)CCC(C)N(c2nnc(C(F)F)s2)C1 82357,C1(CNC(=O)Nc2nc3ccccc3[nH]2)COC2(CCCCC2)O1 82358,C1(C(N2C(c3n(C)ncc3)CCC2)=O)C(C)(C)CCCC1(C)C 82359,C1(NC(CCOCCC)=O)CCOCC1C(=O)N(CCOC)CC 82360,n1(CC(=O)NCC(CC)NC(c2ccc(N)cc2F)=O)cc(C)c2ccccc12 82361,C1(C(N2CCC(CNC(Cc3c(C(=O)OC)c[nH]n3)=O)C2)=O)(CF)CCOCC1 82362,C(=O)(C(F)(F)C(F)F)N1CCC(C(C)NC(=O)CC2CCCOC2)CC1 82363,C(c1cnc(O)nc1O)=CC(=O)NCCC(C)NC(C1SCCS1)=O 82364,N1(C(CCCC(C)=O)=O)CCCC2(NC(=O)CCC3CCC(=O)N3)CC2C1 82365,c1(C(N(C(CNC(C(C)=C(CC)C)=O)C)C)=O)cc(OC)nc2ccccc12 82366,c1(-c2nnc(N(C(C3CCCOC3)C)C)n2C)cccc(F)c1C 82367,c1(N2CC(F)CC(C(=O)NCc3cncc(Cl)n3)C2)ncc2cc(Br)ccc2n1 82368,N1(C(c2c(C)cncn2)=O)CCC(CO)(CNC(c2scnc2Cl)=O)CC1 82369,CCCCCC(O)C(C)C(=O)NCC1(CNC(c2ccnn2CCF)=O)CC1 82370,Cc1cc(C(=O)C(=O)NC2CC2NC(=O)C=CC2CC2)ccc1F 82371,C1(NC(C(=O)NCCC(N)=O)=O)CC(F)(CNC(c2csc(CO)n2)=O)C1 82372,C1(CNC(CC(=C)C)=O)CC(NC(c2cc(CC)n(CCO)n2)=O)C(O)C1 82373,c1(C(N2C(CNC(C(C)(C)O)=O)CCCC2)=O)cccc2nc[nH]c12 82374,c1(C(=O)NC2(CF)CCN(C(c3ncc(CC)nc3)=O)C2)cc2ccncc2s1 82375,N1(C(CN(C)C2CC2)=O)CCOC2(C1)CN(C(C1(C)CCC1)=O)C2 82376,C1(NC(C(CC)C2CCOCC2)=O)CC2(C1)CC(NC(C1CCCC(C)O1)=O)C2 82377,C(CN=c1[nH]c(=NCc2ccc(SC)o2)[nH]c2c1COCC2)(c1ccsc1)OC 82378,CON(CCO)C(=O)C1C2CCC1(c1cccs1)C2 82379,C1(CNC(C(C)CF)=O)CN(C(c2cc(C(F)F)on2)=O)CCC12CCC2 82380,C1(C)(C(=O)OC)CN(C(c2ccc(O)nc2Cl)=O)CC1(F)F 82381,CC(C)C(C(=O)NC1CCN(C(c2cc(C(N)=O)co2)=O)C1C)n1cncn1 82382,C(c1cccc(F)c1)=CC(N1CC(NC(c2cnc(O)s2)=O)C(O)C1)=O 82383,c1(OC)ccc(C(C)CC(=O)NCC(O)CNC(=O)C(C)O)cc1 82384,C(c1cc[nH]c1)=CC(=O)NC1C(CNC(=O)C=CI)C1 82385,C1(NC(C(CSC)OC)=O)COCCC1NC(C1CC(C)(C)C1)=O 82386,C#CCCC(C(=O)NC1(C2CCCC2)CC1)NC(=O)CC12CCCC1C2 82387,C1(C(=O)NC(CC(C)NC(c2cccnn2)=O)C)CN2CCN1CC2 82388,c1(N(C2CCN(C(c3ccc(C)c(F)n3)=O)C2)C)ccc2c(n1)CCC2=O 82389,C1(C)(CC)CCCN(C(=O)CC(C)NC(c2csnc2C)=O)CC1 82390,C(C)(N=c1[nH]c(Cl)ncc1C1CC1)C1N(C(Cc2nnn(CC(C)C)n2)=O)CCC1 82391,Cc1cc2c[nH]nc2cc1C(=O)N(CC(C)(C)NC(=O)C=C1CCCCC1)C 82392,C1(N(C)C(c2cc(S(N)(=O)=O)co2)=O)COC2(CCN(C(=O)C(C)(F)F)CC2)C1 82393,C1(NC(=O)C=CC2CCCO2)CCCCN(C(=O)Cc2sc(O)nc2O)C1 82394,c1(NCCCCOCC)cc(C)c(S(=O)(=O)N2CCCCC(C)(C)C2)cn1 82395,C1(CNC(c2cnns2)=O)CN(C(C2CCCCCCC2)=O)C2CCCC2O1 82396,C12(C(=O)NCC(C)N(C)C(c3cc(F)cc(F)c3)=O)CC3CC(CC(C3)O1)C2 82397,O(C=CC(=O)NCC(C)N(C)C(c1ccn(CC)n1)=O)CC 82398,C1(NC(CCCC=C)=O)CC2CC(NC(c3cnc(N(C)C)s3)=O)CC12 82399,Cc1ccc(F)cc1C(=O)N(CCC(=O)NCC(CNC(N)=O)ON)C 82400,C1(F)(C(=O)NCC(C)(CO)NC(C(CSC)OC)=O)CCCCCC1 82401,C1(NC(CCCOC)=O)CCC(NC(c2cccc(OC(C)C#N)c2)=O)CC1 82402,C(CCCC(=O)NC1CC(=O)N(C(C)C)C1)NC(COCCSC)=O 82403,CC(O)C(C(F)(F)F)NC(=O)CNC(=O)Nc1ccc(C(N)=O)cc1F 82404,C1(C(=O)NCC2CCC2NC(C2(CC3CC3)CCC2)=O)CCC2(CC1)OCCO2 82405,CC(C)CC(C(=O)N1CCCC(O)(CO)C1)NC(=O)CN(C)C(=O)C1CC1 82406,N1(C(C(c2ccoc2)NC(C(OC)OC)=O)=O)CC(O)(C(F)F)C1 82407,c1(C(=O)OC)cccc(N=[N+]=[N-])c1.C12CCN(C1)C(=O)N2CC1CCCO1 82408,C12(NC(c3cc(C#N)sc3)=O)CCN(C(c3cc(Cl)c[nH]3)=O)CC1C2 82409,Cc1c(C(N2CCN(C)CC2CNC(=O)C(O)C(C)(C)C)=O)cccc1CO 82410,C(=O)(CC(C)C(F)(F)F)NCCC(C)NC(=O)CSCc1ncc[nH]1 82411,C1(CNC(Cc2cnn(C)n2)=O)CCCC(NC(c2coc(CO)c2)=O)C1 82412,C1(NC(COC2CCN(C)CC2)=O)CN(C(C2(Cl)CC2(F)F)=O)CC1(C)C 82413,N1(C(CC(C)SC)=O)CC(CNC(=O)CSc2nncn2C)C(O)C1 82414,c1(C(=O)NC(C(C)NC(C2(CSC)CC2)=O)C)cc(Cl)ccc1C(F)F 82415,n1(C2CN(C=O)C2)cc(CCC)nn1.C1(OCC)CCN(C(c2coc(OC)n2)=O)C1 82416,CCC(C)CCC(=O)NC(CC)CC(=O)NC(c1ccc(O)nc1)C 82417,N1(C(C(C(C)(C)C)O)=O)CC2CC1CN(C(c1cc(F)cnc1O)=O)C2 82418,C(=O)(C1=C(NC(C2CCN2c2ncc(CC)s2)=O)CCCC1)OCC 82419,N1(C(C=Cc2ncc(C)[nH]2)=O)CCCC(NC(=O)CCc2ncccn2)C1C 82420,Cc1cc(C#N)ccc1C(=O)NC(C(=O)NCc1c[nH]nc1C(C)C)C1CC1 82421,CC(C)(CCCF)C(=O)NC1CCCCC1CC(=O)NCC1(C)CC2(CCC2)C1 82422,N1(C(CS(=O)(=O)NC)=O)CCC2C(C1)NC(=O)CN2C(=O)CN(C)C(=O)OC 82423,c1(CSCC(=O)NC2COC3(CC3)C2)nc2ccccc2[nH]1 82424,C(C(C(=O)NC1(CCF)CCC1)C(C)(C)C)NC(CCC(C)(C)OC)=O 82425,c1(OC)cc(C2(C(N3CCCC3c3ccc(Cl)c(F)c3)=O)CCCC2)ccc1C 82426,C1(N=[N+]=[N-])(C(=O)Nc2c(C)cccc2F)CCN(C(c2csc(C)c2C)=O)C1 82427,C(=O)(C1CCCc2nncn21)N1CCN(C2CN(C(c3c(C)nco3)=O)C2)CC1 82428,C12(CN(C(=O)Cn3nc(COC)n(C)c3=O)CC)CC3CC(CC(C3)C1)C2 82429,N1(C(Cn2c(C)nc(C)n2)=O)CC(N(C(=O)C(O)C2CC2)C)C(C)(C)C1 82430,N1(C(C(CCCC)C)=O)CCC2(C1)CN(C(c1ccc(C(=O)CC)cc1)=O)C2 82431,c1(C(=O)NCCN(CC(C)O)C(c2nc(OCC)oc2)=O)ccc(N)cc1C 82432,C=CCC(C)C(=O)N(CCCNC(c1ccc(OC)cn1)=O)C(C)C 82433,C(=O)(C(C)N1CC(C)C1)N(CC(=O)NCC=CC)CC1CC1 82434,CC1(C)CN(C2CCN(C3CCOCC3)C2=O)CCC1NC(=O)CC(F)(F)F 82435,C1(CN(C)C(c2cc(CO)n(C)n2)=O)CCN(C(=O)COCC2CCOC2)CC1 82436,CCC(CNC(=O)CCCc1nc(C(C)C)no1)(CC)NC(c1nc(O)sc1C)=O 82437,CC#CCC(C(=O)N1CC(c2ccccc2)C1)NC(C1CC2CCC2C1)=O 82438,C1(CC(=O)NCC(C)(C2CC2)OC)CCN(C(=O)Cc2csnn2)CC1 82439,C1(C(=O)NCCC(O)CNC(=O)C(C2CC2)C2CC2)CCCS1(=O)=O 82440,CCC(CSC)N=c1[nH]c2c(c(=NC3CCC4(CCC4)CC3)[nH]1)SCC2 82441,N1(C(C(C)N(CCC)C(c2cc(Cl)no2)=O)=O)CCCCCC1C 82442,N1(C(C(C)NC(CC)=O)=O)CCN(C(=O)C=CCN(C)C)C(C(C)C)C1 82443,C(=O)(CC(F)(F)CC(=O)N1CCCC1(C)CNC(C1CCC(C)CC1)=O)OC 82444,C1(CCNC(c2cn(C)nc2C2CCC2)=O)CN(C(=O)C=CCO)CCS1(=O)=O 82445,c1(C(CCOCC2CC2)NCC(CC)C)nnnn1CCOC 82446,Cc1cccc(C(=O)NCC2(F)CCC(NC(=O)C(c3ccccc3Cl)C)C2)n1 82447,C12(NC(=O)CCc3ncccn3)CCCN(C(c3cncc(F)c3)=O)CC1C2 82448,Cc1nccc(C(=O)NC(C)CC(C)NC(=O)C(C)Sc2ccccn2)c1C 82449,C1(CNC(c2c(C)cn(C)c2)=O)CN(C(=O)C(N2CCCCCC2)C)CCCO1 82450,N1(C(C2(C)CC2(F)Cl)=O)CCC(C)(NC(c2cccc(OC(F)(F)F)c2)=O)CC1 82451,N#CC1(C(N2CCC(O)(c3nc(C4CC4)no3)C2)=O)CC12CCCC2 82452,N1(C(c2c(C#N)cn[nH]2)=O)CCC2(CCN(C(C3CCCCC(F)(F)C3)=O)C2)C1 82453,n1(CC(=O)OC)ncc2ccc(NCc3ccoc3C(=O)OC)cc12 82454,C1(C(N(C)Cc2ccon2)=O)C2CC1N(C(c1csc(F)c1)=O)C2 82455,Cc1cc(Br)c(S(=O)(=O)NCC2(CO)CC23CCOCC3)cc1Br 82456,c1(NC(CC(C)(C)NC(C(C)=CC(C)(C)C)=O)=O)cnc(F)cc1C 82457,CCCC(C(=O)NC1CCN(C(c2ccc(OC)c(C)c2)=O)C1C)S(N)(=O)=O 82458,CC(CC(=O)NCCc1ncnn1C)C(C)(C)NC(=O)C=CC1CC1 82459,N1(C(c2n(CC)cc(Cl)c2)=O)CCC(CNC(=O)COCC2CCCOC2)C1(C)C 82460,C(C(C)(C)CNC(=O)C(C1CC1)NC(c1ccc(Cl)s1)=O)SC 82461,C1(C(=O)NC(CC)CN(C(=O)C(=O)N(C)C)C)CN(C)CCN(C)C1 82462,Cc1c(C(=O)NCC(C)(C)NC(C2CCCS2)=O)ccc(F)c1F 82463,C12(NC(=O)C(C3(O)CC(C(=O)O)C3)c3cccs3)CCN(CC3CC3)CC1C2 82464,C1(C(N(C)CC2N(C(C3(C)ON=C(C)C3)=O)CCC2)=O)CCCC12CCC2 82465,c1(NC(CC)CNC(c2cc(O)nc(Cl)c2)=O)nc2c(cc1C#N)COCC2 82466,C(N=c1[nH]c(=NCCCCN(C)C)[nH]c2c1SCC2)C1(CO)C(C=C)C1 82467,Cc1cnc(C(=O)NCC2CCN(C(=O)C=CC3CCCC3)CC2)cc1C#N 82468,c1(NC(C2N(C(C(CC)NC(N)=O)=O)CC2)=O)cc(C2CC2)cc(F)c1 82469,c1(C(=O)NC2(C)CC(NC(COCCOCC)=O)C2)cnc2[nH]c(=N)sc2c1 82470,C#CC1(NC(c2ncnc(C)c2C#N)=O)CCCC(C)(C)C1 82471,C12CCCCN1N1CCCC1CC2.CP(C)(=O)COCC1CC(OC)C1.CC=O 82472,C1(C(N(CCCNC(c2cc(CCC)[nH]n2)=O)C)=O)COCC(C)O1 82473,C1(CC(C)NC(C2CCS2(=O)=O)=O)CCN(C(=O)CCc2cccs2)CC1 82474,Cc1ccc(F)cc1C(N1CCCC1CCC(=O)NC1(C#N)CCOCC1)=O 82475,C1(CCC)CN(C(=O)CCC(=O)NCCCOC)CCN1C(=O)C(C)CC(N)=O 82476,c1(OC)ccc(C)c(C(=O)NC2CC2CNC(=O)CC2CCC(C(N)=O)CC2)c1 82477,Cc1nonc1CC(=O)N(CCCn1cc(C(O)C2CC2)nn1)Cc1ccccc1 82478,c1(CN2CCC(C(C)C(=O)N(c3cnns3)C(C)=O)CC2)cccc(-c2cnco2)c1 82479,Cc1cc(C(=O)NCC2(O)CCN(C(c3c[nH]cc(C)c3=O)=O)CC2)ccc1Cl 82480,N(C1CCCn2nccc21)C(c1c(CNC(c2nc(C)c(C)s2)=O)ccs1)=O 82481,CC1(C)CN(C(=O)C2=COCCC2)CCN(C(=O)C2=NNC(C(F)(F)F)C2)C1 82482,c1(N(CCCNC(c2c(C)nc(CC(C)C)s2)=O)C2CC2)ncccc1[N+](=O)[O-] 82483,c1(C(=O)NC2(C)CCN(C(COCCCC)=O)C2)cc(C#N)c(N)cc1O 82484,S(=O)(=O)(c1ccccc1N=[N+]=[N-])NC1CN(C(C)=O)C1 82485,N1(C(COC(CC)(C)C)=O)CC2CCN(C(=O)CC3(OC)CCOCC3)C(C2)C1 82486,C(=O)(CC(C)N(C(N)=O)CC1CCCC1)NCCN(C(C=CCC)=O)CC(C)O 82487,c1(C(=O)NC2CC(NC(C3(CC=C)CC3)=O)C2)nc2ccccc2[nH]1 82488,c1(C(=O)NC2CCCCN(C(C(CCC)OC)=O)C2)coc(=O)c2ccccc12 82489,C(=O)(CCCCCN(C)C(C1CC1[N+](=O)[O-])=O)N1CC(CCC#C)C1 82490,N1(C(c2cnsc2)=O)CCC2(CCCN(C(C3CC34CC(O)C4)=O)C2)C1 82491,c1(C(N2CCC(O)(C(C)NC(c3cccc(O)n3)=O)C2)=O)occ2c1CCC2 82492,CC(C(C)(C)C(=O)N1CCC1C1CCCC1)NC(=O)CC1C=CCC1 82493,C1(NC(CNS(CCCC)(=O)=O)=O)CCN(C(c2ccc(O)nn2)=O)CC1CC 82494,N1(C(CCC(C)N(C2CCCC2)C)=O)CCC2CCC(C1)N2CC(n1cncn1)Br 82495,C(=O)(C1=CCC(C)(C)CC1)NC(C1CN(C(c2cnncc2O)=O)CCO1)C 82496,c1(CNCC2CN(C(C3C(c4n(C)cnc4)C3)=O)C2)cccc2c1OCCN2 82497,N1(C(CCc2n(C)ncc2)=O)CCCC1(C(=O)NC12CC(C1)C2)C(C)C 82498,c1(N(CC(C)NC(=O)OCCCc2csc(C3CCCC3)n2)C)ccccc1 82499,CCCCCCCCC(C)C(=O)N1CC2(CCN(C(=O)C(C)N(C)C)CC2)C1 82500,C(CC(F)F)(C(=O)N1CC=CCO1)NC(c1ccc(CC#N)cc1)=O 82501,C(=O)(N1OC2CCC1CC2)c1c(C)oc(CNC(c2cccc(O)c2F)=O)n1 82502,c1(CCC(=O)NCCC2CCN(c3nc(C4CC4)ns3)C2)nc(O)n[nH]1 82503,N1(C(C2N(C)CCC2)=O)CCOC(C(=O)NC2CCN(CC3CC3)C2)CC1 82504,C1(N(C(C2COC(=O)C2)=O)CC)CCN(C(C2CC(N=[N+]=[N-])C2)=O)CC1 82505,CC1(C)CC(C)(C(N2CCN(C(N)=O)CC2)=O)CN1C(c1cscc1Cl)=O 82506,C(=O)(C1SCCc2ccccc21)N1CCN(C(C=C=C(C)C)=O)C(CCO)C1 82507,C(C)(CC(C)C(F)F)NC(CCCCNC(C1(CC)CC(C)(C)C1)=O)=O 82508,c1(CC(=O)NCCCCNC(CCC(=C)Br)=O)c(F)cccc1C#N 82509,Cc1ccc2[nH]c(C(N3CCCC(N(c4ncnc(=N)[nH]4)CCO)C3)=O)cc2c1C 82510,CCCC(CC(=O)NCCC(C(C)C)N(C)C)NC(c1ocnc1C1CC1)=O 82511,N1(C(C2C(CC)N(C(=O)C(C)OCC3CC3)CC2)=O)CCC(C)CC1C 82512,N1(C(c2ccc(CC)o2)=O)C(CNC(=O)COCc2ccnn2C)CC2CC12 82513,C1(NC(C2CN(C(C)=O)C2)=O)COC2(CCN(C(c3cc(Cl)ccc3N)=O)C2)C1 82514,N1(C(CCC(=O)N(C)C)=O)CCN(C(C2CCC(C(C)(C)O)CC2)=O)CC(O)C1 82515,Cc1ccc(N2CCC(NC(C3(F)CCCCC3)=O)C(O)C2)c([N+](=O)[O-])c1 82516,Cc1ccc(C=CC(=O)N(C2CCCCC2NC(=O)C(F)F)C)c(C)c1 82517,C(C(=O)N(C)CC1CN(C(=O)CC2(O)CCN(C)CC2)C1)(C(C)(C)C)OC 82518,c1(OC)nccc(C(=O)NCCCC(C)NC(=O)CC(O)C(C)C)c1F 82519,C1(C(N2C(CC(=O)NC)CC2)=O)CCCN1C(=O)CCC1CC1 82520,NC(C(=O)NNC(=O)c1ncon1)c1c(F)cccc1Cl 82521,c1(-c2n(C)ncn2)ccccc1CNC(=O)Nc1ccc(F)nc1 82522,c1(C(=O)NC2CC(C(=O)O)CN(C(C(CC(N)=O)O)=O)C2)n[nH]c2c1CCSC2 82523,O=C(NNC(=O)c1c[nH]c(Br)c1)c1cccc(-n2cc(CCCCO)nn2)c1 82524,N1(C(C2(CNC(C(CC=CCC)C)=O)CC23CCC3)=O)CCC(C2=NOCC2)C1 82525,C1(C(=O)NC(CCC#C)=O)CN(C(=O)CCc2nnc(C(F)F)o2)CC1C 82526,c1(CC)ccc(C(=O)N(C2CCN(C(C3CCCC(CF)C3)=O)C2)C)cn1 82527,n1(CCCC)ncc(C(=O)NCC(CC(C)C)NC(c2cnnc(Cl)c2)=O)c1C 82528,C(CO)(CCC(C)C)NC(CONC(C1(SC)CCC1)=O)=O 82529,C(=O)(C1=CC(c2ccccc2)NC(=O)N1)N(CC(=O)O)Cc1cnccn1 82530,C(c1cn(C)cn1)=CC(=O)NCCSCC(=O)N(C)Cc1nc[nH]n1 82531,C1(NC(C)=O)CCCN(C(C2CC(O)(CNC(c3ccn(C(C)C)n3)=O)C2)=O)C1 82532,CC1(CCC(=O)NC2CC(C)(NC(c3csc(C4CC4)n3)=O)C2)CC1(F)F 82533,Cc1cc(Cl)cc(C(=O)NCC(C(C)C)NC(=O)Cc2ccc(F)c(Cl)c2)c1N 82534,C1(=CCC)CCN(C(c2nocc2CC)C(=O)NC(C)C)C1 82535,C1(NC(C=CCN(CC)CC)=O)CC2CN(C(=O)CS(N)(=O)=O)CCN2C1=O 82536,c1(C(=O)OC(c2ccc(Br)s2)C)ccc(C2CCCC2)c(F)c1 82537,n1(CC)cc(S(=O)(=O)N2CC3CN(C(=O)Cc4ccc(Cl)cc4)CC3C2)cn1 82538,N1(CC(CNC(C2CCCN2C(C)=O)=O)OC)CCCC1=O 82539,N1(C(C(c2c(C)cccc2Br)NC(C(COCC)C)=O)=O)CCCCCC1CC 82540,C1(c2onc(-c3cc(C)nn3CC(F)F)n2)C2CN(C(CCC=C)=O)CC12 82541,C12(CNC(C(C)SC)=O)CN(C(=O)Cn3ncn4cccc4c3=O)CC1CCO2 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82806,CC1CC(=O)NCCN1C(=O)CC(C)CNC(c1ccn(C)n1)=O 82807,C(=O)(C(F)C(C)C(F)(F)F)N1C(CNC(CC(CC)c2ccc(C)cc2)=O)CC1 82808,C(CC(=O)N1CCCN(C)C(=O)C1)(C(C)CC)NC(C(CC)n1cncn1)=O 82809,c1(OC)cc(F)c(C(=O)NCC(CNC(=O)C(C)(C)OC)C(F)(F)F)c(F)c1 82810,O=C(CCC(CF)CF)NCC#CCNC(C1CCCCC1C(N)=O)=O 82811,c1(CC)nc(CNCC(N)C(=O)ON(C)C)n(C)n1 82812,c1(CC(=O)NCCCN(C)C(c2nc(Cl)sc2Cl)=O)cccc(C2CC2)c1 82813,C(CCCCCNC(=O)CC(C)c1cnn(C)c1)N(C(=O)Cc1cncn1C)C 82814,c1(N2CCC(C(C)NC(=O)CCN3CCC(F)C3)C2)nc(C2CC2)nc(=N)[nH]1 82815,Cc1[nH]cc([N+](=O)[O-])c(=O)c1C(=O)NC1CCCC(NC(=O)C(C)C(C)C)C1 82816,C1(NC(c2c(CC)scn2)=O)CN(C(=O)CNC(=O)CC(C)(C)C)C2(CCC2)C1 82817,C=C(Cl)CC(C(=O)NCC1(O)CC(C)(C)C1)NC(c1ccc(OC)cn1)=O 82818,N12CC(O)C(O)C(O)C1C2=O.c1(C2C(C(=O)O)(COC)C2)ccccc1 82819,CCS(=O)(=O)C1(CNc2cc(NCC3(C)CCCCC3O)nc(C)n2)CC1 82820,C(=O)(C(C(=O)N1CC(F)(C(N2CCC(F)(C(N)=O)C2)=O)C1)OC)OCC 82821,Cc1ccc(OC(C)C(=O)NC(c2ccccc2)CN(C(=O)CC(C)C)CCl)cc1 82822,C(c1ccc([N+](=O)[O-])s1)=CC(N1CCC(CN(C)C(C2(C)C=CCCC2)=O)C1)=O 82823,c1(N(C)C)ccnc(C(=O)NCC(C)(CO)NC(=O)CC=C(Cl)Cl)c1 82824,c1(C(=O)NCC2C(C)CCN2C(c2ccns2)=O)ccc2c(c1)CCC2 82825,N1(C(C)=O)CCC(N=c2[nH]c3c(c(=NCC4CCC(C5CC5)O4)[nH]2)SCC3)C1 82826,Cc1nnn(CC(=O)N(CCC(C)NC(=O)CC(C)c2ccncc2)C)n1 82827,C(CCCC(CO)NC(=O)C(F)=C(C)C)NC(C=C(C)c1ccsc1)=O 82828,C(=O)(CS(=O)(=O)C1CC1)N(CCOC)CCNC(c1cc(OC)nn1C)=O 82829,C1(CC(=O)NCC2CC(C(=O)N(C3CC3)Cc3ccsc3)C2)CCOC1 82830,C1(C(=O)NCCN(C(=O)CCc2ccncc2)CCCN(C)C)CCOCC1 82831,CC(CCNCCCCCC1OCCO1)CC(C)(C)C 82832,Cn1ncc(C(=O)NCc2nocc2C(N2CC(SC(F)F)C2)=O)c1N 82833,Cc1cnc(Cl)c(C(=O)NC(C2CN(C(C3(C)CC3(F)Cl)=O)CCO2)C)c1 82834,N1(C(C(CC)(C)CC)=O)CCCCC(CNC(c2cnc(SC)s2)=O)CC1 82835,C1(C(=O)NCC2C(NC(C3CC4(CCOC4)C3)=O)CC2)CN2CCC1CC2 82836,C1(C2CC2)(C(=O)Nc2c(C)noc2CC2CC2)CN(C(C2CC23CC3)=O)C1 82837,c1(CC(N2CCCCC2Cn2cc(CCCO)nn2)=O)cccnc1Cl 82838,N1(C(C(N2CCOCC2)C)=O)CC2(CC(NC(=O)C(C)(O)C3CCC3)C2)C1 82839,c1(C(=O)NCCCC(C)(C)NC(C(C)n2ccnc2)=O)ncc(F)cc1F 82840,CC(C)CCC(C)NC(=O)C(C)(C)C1CCCN1C(=O)CCN=[N+]=[N-] 82841,c1(C(=O)NCC2C(NC(C3(C)CC3(F)F)=O)CC2)cnc(Cl)c(N)c1 82842,N1(CCc2scc(C)n2)CCOCC1c1cccs1 82843,Cc1nn(C)c2c(NCC3COCC3O)nc(=NCCC(F)F)[nH]c12 82844,CC1CN(c2cc(C(N3CCC=CC3CO)=O)ccn2)CCO1 82845,c1(C(=O)OC)cc(C)n(CC(=O)NCC(C)(O)CNC(=O)Cc2cncnc2)n1 82846,C12(C(N(CCO)Cc3c(C)cccc3)=O)CCC(C1)CC21NC(=O)NC1=O 82847,N1(C(C(CNC(C)=O)(C)C)=O)CCC2(CC1)CN(C(c1[nH]cc3c1CCC3)=O)C2 82848,Cc1nc(CC(=O)NC(C(=O)NCC2CCCSC2)c2cccs2)n[nH]1 82849,N1(C(C(C=C)OC)=O)CCN(C(C2CCCN(C(=O)CCC(F)F)C2)=O)CC1 82850,C1(NC(C2N(C(C)=O)CCC2)=O)CN(C(c2cnccn2)=O)CCC1C 82851,c1(CN(C)C)ccoc1C(=O)N(CCCCNC(=O)C=CC(F)F)C 82852,CCCC(CNC(c1n[nH]c2c1COC2)=O)C(=O)NC1(CC)CC1 82853,C1(NC(c2ccnnc2O)=O)C=CCN(C(c2ccc(CO)cc2)=O)C1 82854,C1(C#N)(C(=O)NC2CCCN(C(CSCC(C)C)=O)C2)CCOCC1 82855,C(=O)(CCCCCCCCCO)N(C1CN(C(C2CC3CC2CC3(F)F)=O)C1)C 82856,N1(C(C(C)SC)=O)CCCCC1C(=O)NCC1CC1(C)C 82857,C#Cc1ccc(C(=O)NC2CC23CC(NC(=O)C(O)CC2CCCCC2)C3)nc1 82858,CN1CC(NC(C2CN(C(c3ccccn3)=O)CCO2)=O)CC1CO 82859,C1(NC(C(C2CCC(C)CC2)CC)=O)CCCN(C(=O)CC(=O)NC2CC2)CC1 82860,N1(C(CN(C)CC)=O)C2CCC1CN(C(=O)C(C)Cc1cnc[nH]1)C2 82861,CC1=NNC(=O)C1CC(=O)NC(CO)C(C)NC(=O)Cn1c(C)csc1=O 82862,C12(C(N(C(C)C)CCN(C)C(C3CCCC3C)=O)=O)CCOC1CCOC2 82863,C1(=CC(=O)NC2CCCC(NC(=O)Cc3ccoc3)C2)CN2CCC1CC2 82864,C(CC(=O)Nc1cc(O)cc(F)c1)(C(F)F)NC(c1n(CC)nc(C)c1)=O 82865,C1(NC(c2ccc(OCC)cc2)=O)CCC12CCN(C(c1sccc1Br)=O)CC2 82866,C=CC(C)(CC)C(=O)N1CCN(CCn2cc(C(C)(C)C(N)=O)nn2)C(=O)C1 82867,c1(OC)ccc(C(=O)NCC2(CNC(=O)Cn3nccn3)CCC2)n2nccc12 82868,C(=O)(C1CCCc2ccccc21)NC(C)CNC(=O)C(C1CCC(=O)N1)C 82869,c1(C(c2cn(CCC(=O)N(C(C)(C)C)CCF)nn2)C)cccc(C(C)(C)C)c1 82870,C(=O)(CC(C(F)(F)F)NC(c1ccc2c[nH]nc2c1)=O)NCCC 82871,C1(NC(C(C)(c2ccccc2)OC)=O)CCN(C(=O)CN2CCC2)CC1C 82872,C12(CNC(C3(CC#C)CCOC3)=O)CC(CO1)N(C(c1cc3n(n1)CCC3)=O)C2 82873,C=C1CC(C(=O)NC(C2CCCC2)CNC(=O)CN2CCCC2C2CC2)(CO)C1 82874,C1(C(N2C(C)(CNC(=O)COc3ccc(F)nc3)CCC2)=O)CCCCNC1=O 82875,c1(NC(CCCNC(CCC(=O)OC)=O)=O)c(OC)cccc1O 82876,C1(C)(C(N2C(C=C)CC2)=O)CCN(C(C2CCCCC2C(=O)OC)=O)CC1 82877,O(N=C1CCCCCC1)CC(=O)NCC(CNC(C(C)OCCC=C)=O)F 82878,N1(C(C2(CC)CC2(F)F)=O)CCN(C(c2cc(-c3ccccn3)no2)=O)CC1 82879,N1(C(c2ccc(C(C)=O)c(F)c2)=O)CCN(C(=O)Cn2cnnc2O)C(C)C1C 82880,C(=O)(CCCS(C)(=O)=O)NC(C1CCCN(C(c2cccc(C)c2N)=O)C1)C 82881,CC(C)S(=O)(=O)CC(=O)NC1(CNC(=O)C(=O)Nc2ncc[nH]2)CCCCC1C 82882,N1(C(C2(COC)CCOCC2)=O)CCCC(CNC(c2cc(OC)cs2)=O)CC1 82883,Cc1onc(CO)c1C(=O)N(CC(C)NC(c1ccc(C(C)(C)C)nc1)=O)C 82884,C1(CCOC)CN(C(c2csc(-c3ccncc3)n2)=O)CCN1C(=O)C(N)=O 82885,N1(C(C2C(OC)(OC)CC2)=O)CCC(F)(CNC(=O)CCc2nc(CO)no2)C1 82886,c1(C(=O)NCCCCCNC(c2ccc[n+]([O-])c2)=O)ncc(F)cc1F 82887,Cc1nccc(C(N2CCCCC2CCC(=O)N(C2(C)CC2)C)=O)n1 82888,C(C)(C(=O)NC1CC(F)(CNC(C2(N(C)C)CCCOC2)=O)C1)(C(C)C)OC 82889,C1(C(=O)NC2C(C)CN(c3nnc(C#N)s3)CC2)CN2CCN1C(C)C2 82890,C1(C(=O)NCCN(CC(F)F)C)CC2(CCC2)CN1C(=O)CC1CCCO1 82891,c1(C(=O)NCCNC(C(COC(C)(C)C)N(C)C)=O)cc(Br)ccc1O 82892,C(c1cn(C)cn1)=CC(=O)NC(CCOC)CNC(=O)CSCCC(F)(F)F 82893,CC1CN(C(=O)CC2CCN(C)CC2)CCC1N(C(=O)Cc1ccnn1C)C 82894,C1(CNC(CCC(=C)C)=O)CCCN(C(c2cc(NC(C)=O)cnc2C)=O)CC1 82895,N1(C(CNS(N(C)C)(=O)=O)=O)CCN(C(=O)C(C)(O)C2CC2)CC(CO)C1 82896,S(=O)(=O)(c1cc(C(F)(F)F)ccc1NCCF)NC(c1cc2ccccc2o1)C 82897,c1(CNC(CCC2(C)CCN(C(C3C(C)(C)C3)=O)C2)=O)ccnc(C#N)c1 82898,C(CCC(C)CO)NC(C1(NC(CC)=O)CCSC1)=O 82899,C=C1CC(C(=O)Nc2cc(C(=O)OC)no2)N(C(=O)Cc2ccc(Br)cc2)C1 82900,Cc1nnc2n1CC(C(N1CCOCC(NC(=O)Cc3ccoc3)C1)=O)CC2 82901,Cc1cc(NC(c2cnn(CCO)c2C(F)(F)F)=O)ccc1NC(=O)C(C)O 82902,C(=O)(C1COc2ccc(Cl)cc21)N1CC(NC(C(C)(C)C2CC2)=O)C(C(F)F)C1 82903,C1(C(c2ccsc2)CNC(C2CCC2)=O)CCCN1C(=O)CCc1ccoc1 82904,n1(CC)nccc1C=CC(=O)N(C(C)CN(C)C(c1snnc1C)=O)C 82905,c1(C(N(CC(C2CC(F)(F)C2)O)C)=O)ccc(N)c(Cl)c1 82906,c1(C(=O)NC2CC2C(=O)Nc2ncc(F)cc2Br)cc(Cl)c(Cl)cc1F 82907,C(=O)(CC(F)(F)C(F)F)N(CCCCC1CN(C(=O)CNc2ccc(Cl)cn2)C1)C 82908,N1(C(c2ccc(OCCN(C)C)cc2)=O)CCN(C(=O)C=C2CCC2)C(CF)C1 82909,Cc1nc(-c2cccs2)sc1C(N1CCCC1C(C)(C)NC(=O)COCCF)=O 82910,CC(C)C(O)C(=O)N1CC(C(F)Cn2cc(Cn3cccc3)nn2)C1 82911,c1(CN2CC3C(C(N4CCC(C)CC4)=O)(C3)C2)cc(F)ccc1F 82912,c1(C(N2C(CN(C(C3(CC(C)C)CC3)=O)C)COCC2)=O)nccc2cc[nH]c12 82913,c1(C(N(C)CC2C(C)OCC2)=O)c(CNC(C2SCCS2)=O)nnn1C 82914,C1(CNC(c2cccc(C)c2)=O)CN(C2CCc3ccccc32)C1 82915,C1(C(=O)NCC(C2CCCCC2)NC(=O)C2=CCCC2)CCC(F)(F)CC1 82916,c1(CC)ccc(CNC(=O)CC(C)NC(C2CCOC2C(C)C)=O)cc1 82917,CC1(NC(=O)COC2CCOC2)CC(C(=O)NC(c2csc(O)n2)COC(C)C)C1 82918,CC1CC=C(C(=O)NCc2cc(C(=O)NCC(C)C(C)(F)F)n[nH]2)CC1 82919,c1(CC)ccc(F)cc1C(=O)NC(C(C)NC(=O)CN1CCS(=O)CC1)C(C)C 82920,C1(NC(CCC(=O)OCC)=O)CCCC12CCN(C(C1CCC1(C)C)=O)CC2 82921,Nc1cc([N+](=O)[O-])ccc1C(=O)NCC1CCCN1C(=O)CC1CCC(=O)N1 82922,c1(CCC)c(C(N2CC(NC(C3CCCSC3)=O)C(CO)C2)=O)nnn1CC 82923,c1(N2CCSCC(C)C2)nc2ccsc2c(=NCC2(C)CS(=O)(=O)C2)[nH]1 82924,C1(CC)CN(C(c2ccnc(F)c2F)=O)CCN1C(=O)Cc1ccccc1OC 82925,c1(N2CC(C)C(NC(=O)CC3CC(F)C3)CC2)ccc(Br)cc1[N+](=O)[O-] 82926,N1(C(c2ccncc2N(C)C(C)C)C(=O)NC)CC2CC(OC)C(C2)C1 82927,N1(C(c2nn(C)c(=O)cc2)=O)C2CCC1CN(C(c1ncc(Cl)c(N)c1Cl)=O)C2 82928,N1(C(C2(COCC)CC2)=O)CCCC(CCNC(C2CCCC(O)C2)=O)CC1 82929,c1(CC(=O)NCC(C2CCOC2)NC(CC2(OC)CCCC2)=O)ccncc1F 82930,CC1CN(C(=O)Cc2ccon2)CC2(CCN(C(C3CC(C)(F)C3)=O)C2)O1 82931,c1(C(=O)OCC)ccc(N2CCC(NC(=O)Cc3ccn(C(C)C)n3)C2)nc1C 82932,C1(NC(C=CS(C)=O)=O)C2CC(O)C1N(C(=O)CCCc1ccccc1)C2 82933,Cc1cc(=NCC2CCCC(C)CC2)[nH]c(=NCCc2cccc(N)c2)[nH]1 82934,CCCC(CC)CCC(=O)NC1CCC(NC(c2sccc2OC)=O)CC1 82935,N1(C(C(C)OCC2CC2)=O)CCC(NC(=O)CCC2CCOCC2)C(CO)C1 82936,CC1(C)CC(CNC(C2CC23CC(O)C3)=O)CN1C(=O)CCC1CCC1 82937,c1(C(=O)NC2(CN(C(=O)CCC(N)=O)C)CC2)cnc(O)c2cccnc12 82938,Cc1cc(C)c(CC(N2CCOC(CCNC(C3CCC3)=O)C2)=O)c(C)c1 82939,C1(CC(=O)NCc2[nH]nnc2C)(OC)CN(C(=O)C(c2cnn(C)c2)=O)C1 82940,CC1CCCC(C(=O)NCc2nocc2C(=O)NCCC(C)C(F)F)C1 82941,c1(C(=O)NC(C(=O)N(CCNC(c2c(C)occ2)=O)C2CC2)C)cccc(Cl)c1 82942,C1(C(=O)NCc2cncc(C)c2)CCN(C(=O)C(C)OCC(C)C)CC1(C)C 82943,C1(CC(=O)OC)(NCC(C)(C)c2nn[nH]n2)CCN(C)C1 82944,C(=O)(C(C(C)=Cc1ccccc1)N1CCC(OC)(OC)C1)NCCCOC 82945,CCC(CC(=O)NCC(O)CN(C)C(c1ncoc1-c1cnn(C)c1)=O)C(C)C 82946,c1(CC(=O)OC)ccccc1C(=O)NCC1C2CC2CN1C(C1C=CCC1)=O 82947,c1(CNC(c2cc(CC)oc2)=O)ccc(NC(C2C(OC(C)=O)COC2)=O)cc1 82948,N(C(=NCCN(CC(F)(F)F)C(C)C)NCCN1CCCC1)C1CCC(C)CC1 82949,C1(CNC(CCN(C(=O)CCOC2COC2)C)=O)(CO)CCCO1 82950,C1(CC)CCCC1C(=O)N(C1CC(C(=O)NCCCCC(=O)NC(C)(C)C)C1)C 82951,C1(C)(C(=O)NC(C)Cc2nncn2C)CCN(CC2CCCOC2)CC1 82952,N1(C2CCN(CC)C2=O)CC(NC(c2ccn(-c3ccncc3)n2)=O)C(C)(C)C1 82953,c1(C(=O)OC)ccc(CNC(=O)N(CC(c2cccc(OC)c2)O)C)cn1 82954,C12(CN)CC(C1)C(NC(c1cncc(-c3cc[nH]n3)c1)=O)CO2 82955,C=CC(O)C(=O)NCCCCN(C(=O)CN1CCC(OC)C1)C 82956,c1(N(CC(CC)C)C)nc(NCc2c(C)nc3ccccn23)c2ncn(C)c2n1 82957,c1(C(=O)NCC2(C)CCCN2C(c2ncccc2Br)=O)n[nH]c2c1COC2 82958,C1(NCC(c2ccc(F)c(Cl)c2)O)COCC1C1CC1 82959,C1(NC(c2c(CC)nco2)=O)CCC2CCN(C(C3(C)CC(C)C3)=O)C1C2 82960,c1(COC)nccc(=NCCN(C(=O)CC2Cc3ccccc3O2)C(C)C)[nH]1 82961,c1(C(C)CC(=O)NC(C2CN(C(C3(O)CCSCC3)=O)C2)C)c(F)cccc1F 82962,C(=O)(C1=Cc2ccccc2C1)N1CCC(C(C)NC(C2C3CC3C3CC23)=O)CC1 82963,N1(C(C(C2CCC2)OCC)=O)CC2(CCCCN2C(c2ccnc(S)c2)=O)C1 82964,CC(C)(C)CC(F)C(=O)N1CCC(NC(c2cc3cnccc3[nH]2)=O)C(F)C1 82965,CCCC(C(=O)N1CCC(C)N(C(c2cc(C)c(F)cc2F)=O)CC1)S(N)(=O)=O 82966,N1(C(C)=O)CCN(CCN(C(=O)C(F)OC(F)(F)F)C)CC1.c12ccc(cc1)[nH]2 82967,Cc1coc(C)c1CNC(=O)C(=O)NCC1CCCC1CC(C)C 82968,Cc1cc(=NC(=O)c2ccc(F)c(C(F)F)c2F)[nH]n1-c1ccc(Cl)c(F)c1 82969,Nc1sc2ccccc2c1C(N1CCCOC(CNC(c2cc(Cl)c[nH]2)=O)C1)=O 82970,CCC(CC(C)C)C(=O)NC1CC(F)(CNC(c2cc3ccccc3o2)=O)C1 82971,CCC(CC)(C(=O)N1CCC(NC(=O)CCC(C)(C)F)C(C)C1)OC 82972,c1(OC)cc(C)cnc1C(=O)N(C)CC1C2CN(C(C3CC3C)=O)CC12 82973,c1(C(N(C2CCN(C(c3ncoc3CC)=O)C2)CCC)=O)cnc(C(F)F)cn1 82974,CCCC(O)CC(=O)N1CCOCC1CNC(c1sc(C)nc1CC(C)C)=O 82975,C1(C(=O)NC(C(=O)NC2CN(C(C)C)C(=O)C2)C2CC2)CN(C)CCN1C 82976,CC1CN(C(=O)C2=CCC(NC(=O)CCC(F)(F)F)C2)C(C)C1C 82977,Cc1cccc(CN2CCCC2CCNC(c2csc(-c3ccccc3)n2)=O)n1 82978,Cc1nc(-c2ccccc2)ncc1C(N1CC(O)(CN(C(=O)C(C)C#N)C)C1)=O 82979,c1(OC)ccc2[nH]nc(C(=O)NC3(CNC(c4cncs4)=O)CC(OC)C3)c2c1 82980,C(=O)(C(F)C(=O)NCC(CC)NC(=O)CCCc1cc(C)no1)OCC 82981,CCC(C(=O)NC1CC(F)(CNC(=O)C(C)CC2CC2)C1)OC 82982,C(C)(C(=O)NCC(=O)N(C)O)(C1CCC1)NC(CCOCC)=O 82983,CCS(=O)(=O)C=CC(=O)NCC1CC2CCC(C1)N2C(=O)CCC=C(C)C 82984,C12(C(N3CC(CNC(Cc4c(C)n[nH]c4)=O)C(C)C3)=O)CCC(CC1)CC2 82985,c1(NC(=O)Nc2cn(C(C(=O)OCC)(C)C)nc2)ccc(C)n1C 82986,C1(CN(C(c2[nH]cc(C(=O)OC)c2)=O)C)CCCCN1C(C1CC1C)=O 82987,C1(NC(=O)C=Cc2cnccn2)CS(=O)(=O)CC1NC(c1cc(Cl)ccn1)=O 82988,C1(C(N(C2CCN(C(C(COC)(F)F)=O)CC2)C)=O)CSc2ccccc2O1 82989,C1(C(=O)NCC2C(C(N3CCC(C(C)C#N)CC3)=O)C2)CC12CCOCC2 82990,Cn1cnc2nc(=NCc3nncs3)[nH]c(NCC3C4CCCCCC34)c12 82991,C=C(Cl)C(C)(C)C(=O)N1CC(NC(=O)Cc2cc(OC)ccc2Cl)C2(CC2)C1 82992,CC(C)CC(C(=O)N(C1CCCN(C(c2cn3ccnc3s2)=O)C1)C)C(C)C 82993,C12(C(=O)Nc3cccc(-n4ccnc4O)c3)CCCC1C2(F)F 82994,C(=O)(N=c1[nH]onc1C(C)(C)C)Nc1ccc(COC(=O)NCC)cc1 82995,C(CCCCCNC(c1ccc[n+]([O-])c1)=O)NC(c1ccsc1)=O 82996,C12CC(CN1CC1C3CC4C(C3)C14)SC1=CC=C21.c1(OC)cnc(-c2cccc(O)c2)nc1 82997,C1(N(C(C(C)N=[N+]=[N-])=O)C)CCCN(C(=O)C(c2cncnc2)C)CC1 82998,C12(NC(c3cc(=NC)[nH]cc3)=O)COCCC1CN(C(c1c[nH]cc1Br)=O)C2 82999,C(CCCCC(=O)N1CC2(CC(NC(=O)C(n3cc(C)cn3)C)C2)C1)SC 83000,C1(C(=O)NC2(CC=C)CCCCC2)CN(C)CCN1C(c1ccc(F)c(O)c1)=O 83001,C1(OC)CC(NC(C2(C)CCN(C)C2=O)=O)CN(C(=O)C(C)(C)c2cc[nH]n2)C1 83002,c1(OC)cc2ccc1C(=O)NCCCO2.C(=O)(CCn1cnnn1)NCC1CC1 83003,C(CC1CC1)(C(=O)NC(CC1CCCC1)C(=O)N1CCC(N2CCC2)C1)OC 83004,Cc1cc(CC(N2CC3CCC3(C(=O)NC(c3cnn(C)c3)C)C2)=O)cc(C)c1 83005,C1(NC(CC(=O)OCC)=O)CN(C(=O)C(c2cnn(C)c2)O)CC1C1CC1 83006,CC(CC(=O)c1ccc(F)cc1)C(=O)NC(C)(C)C(=O)N(C1CCCC1)C 83007,c1(C(N(C2CN(C(c3cc(C)no3)=O)CC2F)C)=O)c[nH]c2cnccc12 83008,c1(NC2CC3CN(C(c4cc5sccc5[nH]4)=O)CC32)nc2ccccc2s1 83009,C1(NC(c2c(C)cc(SC)s2)=O)CN(C(c2n[nH]c(C)n2)=O)CC(C)(C)C1 83010,c1(OCC)cc(C(=O)NCC(CNC(=O)CSc2ccncc2)CO)cc(F)c1 83011,c1(OC)c(Br)cccc1S(=O)(=O)N1CCC(NS(C)(=O)=O)C1 83012,C12(C(=O)NCCN(C(C34CCCC3C4(F)F)=O)CC)CCCC1CC(=O)C2 83013,C1(C)(CC)CC(NC(c2cc(F)ccc2F)COC)CCO1 83014,n1(CC)ncc(Cl)c1C(=O)Sc1ccc(Br)s1.N12CCCC1(C)C2 83015,Cc1ccc(C(=O)NC2CCC(C)N(C(C3CC4(C3)CC(O)C4)=O)C2)cc1C#N 83016,C1(C(N2CCC(C(C)NC(Cc3c(C)nc[nH]3)=O)CC2)=O)OCCOC12CCC2 83017,N1(C(c2c(C)c[nH]n2)=O)CCC2(CCC2)C(CNC(C2CCOC2)=O)C1 83018,c1(C(=O)NCC2(C)CCC(NC(c3cc[n+]([O-])cc3)=O)C2)cnc2n1CCC2 83019,c12nc(C)c(s1)CC(=O)NC2.C(C(C(C)C)NC(C1CC1CF)=O)CC(=C)Cl 83020,CC1C(=O)N(C)CCN1C(=O)C(C)(C1CC1)N(C(=O)CCCC1CCCO1)C 83021,Cc1cc(N2CCCCC2CCNC(=O)Cn2nccn2)cc(C#N)c1[N+](=O)[O-] 83022,CCCC(C(=O)NC(c1ccccc1)C1CC1)N1CCCC1CCC 83023,c1(CC)cc(NC(CNC(=O)CCCCNC(N)=O)C2CCC2)ncn1 83024,c1(-c2n(C3C(C)CCCC3C)nc(-c3ccncc3)n2)ccc2cccnc2c1 83025,C1(NC(C2C(NC(C(CO)OC)=O)CCO2)=O)C=C(C)CCC1 83026,N1(C(C(CC)N(C)C)=O)CCN(C(c2ncoc2C2CCCO2)=O)CC(C)(C)C1 83027,c1(C(CC)NC(=O)CCN(C(=O)CC2CC(C)C2)C2CC2)cccnn1 83028,CC#CC1CCN(C(c2cc(C(=O)NCC3CC3CCC)nn2C)=O)C1 83029,Cc1cc(O)ncc1NC(C1(C)CC(O)CN1C(=O)C(C)C(F)(F)F)=O 83030,c1(OC)ccc(C(=O)NC(C2CCCN2CCc2ccccc2)C)cc1 83031,C1(CNC(=O)CCc2nc[nH]n2)CCCCC1NC(=O)CCc1cn[nH]c1 83032,N1(C(C(=O)NCc2nnn(C)n2)c2cncs2)CCCc2occc2C1 83033,N1(C(=O)CC2CC2)CCCCC1C1CCCN1C(=O)Cc1ccccc1 83034,C1(CCNC(C(C(C)C)OC)=O)CCCN(C(c2c(C)noc2N)=O)CC1 83035,CN1C2CCCC1CC(NC(c1ccc(Cl)c(F)c1N)=O)C2 83036,N1(C(=O)NCC(CN=[N+]=[N-])NC(C)(C)C)CC2(CNC(=O)C2)C1.C1(=O)CCN1C 83037,C1(F)(C(=O)NCCOCCC(=O)NCc2nc(C)[nH]n2)CCCCCC1 83038,C(=O)(CC(C)(C)COC)NCC1N(C(c2cc(CCC)no2)=O)CC(OC)C1 83039,C(=O)(C(C)CC(F)F)N1CC(C(C(N2CC(O)C(O)C2)=O)OC)C1 83040,Cc1ccc(C(N2CC3CCC2C3NC(C2(C)CC2(F)F)=O)=O)cc1OC(F)F 83041,N#Cc1ccc(S(=O)(=O)N2CCOC3(CCOC3C)C2)cc1NCC1CC(F)C1 83042,c1(C(N2C(C)CC(NC(CN(CC)CC)=O)C2)=O)cc2cccnc2s1 83043,N1(C(=O)OC)CC(OC)CC1C(N1CC(C)(NC(c2ccc(C)cc2)=O)C1)=O 83044,C1(C(=O)NCC2C(NC(c3c(F)cncc3Cl)=O)CC2)COCCC1(F)F 83045,N1(C(C2C(C)C2C)=O)CCCCC2(CCN(C(C3CC(=O)NC(=O)N3)=O)C2)C1 83046,N1(C(c2c(CC)nn[nH]2)=O)CCOC(C(=O)NCc2nc(C)cs2)CC1 83047,C(CC(CC)C(=O)N(C(CNC(=O)CSCCN(C)C)CC)C)=CC 83048,C1(NC(C2C(OC)CCC2)=O)CC2CCC(C1C)N2C(c1cc(C)ncn1)=O 83049,C1(NC(CC=C)=O)CC2(C1)CC2NC(=O)C(c1ccc(Cl)s1)C 83050,C1(C(=O)NCCCCC2C(C)C2)CN(C(=O)CC2CCCC(=O)C2)CC(C)(C)C1 83051,N1(C(C2(OC)COC2)=O)CCN(C(=O)CNC(=O)C(F)(F)F)C2(CCC2)C1 83052,N#Cc1cccc(I)c1NC(C1CCCCC1NCc1ccc(CO)o1)=O 83053,c1(Nc2scc(CC(=O)Nc3ncc(C)nc3Br)n2)ncnc2cccnc12 83054,c1(C(C)NCC(=O)NCc2ccc(OC(F)F)cc2)ccc(I)cc1 83055,c1(C(=O)NCC(C)CN(C(=O)CN2CCSCC2)C)conc1C1CCCO1 83056,c1(C(=O)OC)c(CSc2noc(C)n2)ccn1C 83057,Cc1c(F)ccc(C(=O)NCC2(O)CCN(C(=O)C(C)C3CCC3)C2)c1C#N 83058,Nc1ccc(C(=O)N(CCC(=O)NCC2CCSC2)CCO)nc1 83059,C1(C(C)C)CC(N=c2[nH]c3c(c(=NCC4(CCCO)CC4)[nH]2)COCC3)CCO1 83060,Cc1ccnc(C(=O)NC2CC(=O)N(C3CN(C(=O)C(C)n4ccnn4)C3)C2)n1 83061,C1(C(CNC(C(CC)C)=O)C)CCN(C(c2[nH]nnc2C(=O)OCC)=O)CC1 83062,N1(C(CC)=O)CCOCC2(COCCN2C(=O)C2CCCn3c(Br)cnc32)C1 83063,C(=O)(C(C)(C1CCC1)NC(c1c(SC)con1)=O)OC 83064,C1(C(=O)NCc2c(C)nccc2)C2CCN(C(=O)CCc3conc3C)CC12 83065,c1(C(=O)NCCC2N(C(c3c(=N)[nH][nH]c3)=O)CCC2)cc(O)nc2ncccc12 83066,c1(N(CC)C)ccc(CN2CCN(C(c3cc(COC)nn3C)=O)C3CC23)c(O)c1 83067,C1(NC(CC)=O)COCCC1CNC(c1cccnn1)=O 83068,c1(OC)cc(O)c(C(N2CCC3CN(C(c4ccsc4Cl)=O)CC23)=O)cc1OC 83069,C(=O)(C(F)(F)C(O)CC)NCC(CC)NC(=O)Cc1sc(C)nc1C 83070,C12(CNC(Cc3c(OC)cccc3Cl)=O)CCCC1CN(C(c1nc[nH]n1)=O)C2 83071,N1(C(=O)CSC2CCCCO2)CC2CC(C1)CN(C(c1coc(C(F)F)c1)=O)C2 83072,Cc1cc(N)c(C(=O)NC(CO)C(C)NC(C2C3CC4C(C3)C24)=O)c(F)c1 83073,C(=O)(C1CCCc2cncn21)NC(C(C)C)CCNC(c1c(O)cccc1Cl)=O 83074,c1sc(C(=O)OCC(C)OC(=O)C(C)N(C(=O)NC(C)(C)C)CC)cc1C 83075,c1(C(=O)NCC(CC=C)NC(C2CS(=O)(=O)C2)=O)cnc2c(F)cc(C)cc2c1 83076,CCCC(C(=O)N1CC(N2CC(F)C2)C1)NC(=O)C(C)c1cccs1 83077,C1(CCNC(CCOCCCNC(C2C(N(C)C)CCC2)=O)=O)NC(=O)NC1=O 83078,C1(F)(CNC(C(C)(C)OC(C)C)c2nnnn2CC2CC2)COCCOC1 83079,C#Cc1cc(C(=O)NCC2CC(C)N(C(c3ccc(Cl)nc3O)=O)C2)ccc1C 83080,CC(=O)CCCC(C)C(=O)N1CCC(C)C1C(N1CC(C)(C)C1)=O 83081,C1(C(=O)NC2C(NC(c3cccc(OC)n3)=O)CCC2)CC12CCC(F)(F)CC2 83082,C1(N(C)C(C2CCCOC2)=O)CCCN(C(=O)C(C)(C)c2ccno2)CC1 83083,c1(C(=O)NC2C(CN(C(=O)C(=CC3CCCCC3)F)C)CCC2)cccc(N)c1 83084,Cc1cc(C#N)ccc1C(=O)NC1(C(=O)NC23CCC(C2)OC3C)CCSC1 83085,C1(CC(N2CC(C(=O)OCC)OCC2)=O)COC2(C1)CN(C(=O)OC(C)(C)C)C2 83086,C(=O)(C(C)CC(C)(F)F)N1C2CN(C(C3(C#N)CC(=C)C3)=O)C(C2)C1 83087,C1(O)(CC)CCN(C(c2nc[nH]c2C(F)(F)F)=O)CC1 83088,C(=O)(C1CC(=O)c2ccccc21)NCCC1CCN(C(c2c(C)scc2)=O)CC1 83089,N1(C(CC(C)F)=O)CC2(CCOCC2)CC1CNC(=O)Cc1ccon1 83090,C1(OC)(CNC(=O)CC2C(NC(=O)CN3CC(C)(C)C3)CC2O)CCOC1 83091,N1(C(C(CCCNC(c2cc(C)nnc2)=O)(C)C)=O)CCC2CCC(O)C1C2 83092,CC1(CN=c2[nH]nco2)CCN(C(=O)C=CC(N)=O)C1 83093,C1(C(N2C(C)(C(=O)NCCNC(=O)NC)CCC2)=O)CC2(CCC2=O)C1 83094,N1(C(C(C)CC2CCC2)=O)CC2(C1)CN(C(=O)CC1(C)CC1(F)Cl)C2 83095,C(CCCCC(=O)NCC1CN(C(c2ocnc2C(C)C)=O)CCO1)OCC 83096,C12(C(=O)NC(CC)C(=O)OC)CC(CN(C(C3CC(=O)C3)=O)C1)C2 83097,c1(CC(N2C(CCC(=O)NCc3cc(F)ccn3)CCC2)=O)ccc(Cl)cc1Cl 83098,N1(C(C(C)c2ncco2)=O)CCN(C(c2cnnn2C)=O)CC1C 83099,N1(C(C2CC(SC)C2)=O)CC(C)CC1C(=O)NCc1nonc1C 83100,C1(F)(CNC(=O)COCC2CCC2)CC(CNC(c2cnn(CC3CC3)c2)=O)C1 83101,C1(C2N(C(Cn3ncc(CC)c3)=O)CCC2)CCN(C(C2CC2C(F)F)=O)CC1 83102,C1(CC)(CC)CC(NC(=O)CC(C)c2ccco2)CN1C(=O)C(C)N1CCC1 83103,c1(C(=O)NCc2ccc(F)cn2)ccc(-c2ccnnc2)c2cc[nH]c12 83104,C1(NC(C2CN(c3nncs3)C2)=O)CCN(C(=O)Cc2csc(Cl)n2)C1 83105,C(=O)(C#CC1CCCCO1)NCCCN(CCCNC(C(F)=C(C)C)=O)C 83106,c1(SCc2cccc(NC(c3ccc(F)cc3)=O)n2)c(F)cncc1Cl 83107,N1(C(C2(CC)CC2)=O)CCC2(CCOC2)C(CNC(c2ccnnc2S)=O)C1 83108,c1(OC)cc(C(N2CCCC2CCNC(=O)CC2COCC(C)O2)=O)n(C)n1 83109,c1(C(N2CCC(CC)(NC(=O)CC34CC(C3)C4)CC2)=O)noc2c1CCCC2 83110,C=CCC(CC=C)C(=O)N1CCN(C(C2CCCCN2CC(F)F)=O)C(C)C1 83111,O=C(C1=COCCO1)NCC12CC(C1)C(NC(c1ncccc1F)=O)CO2 83112,C1(C(=O)NC(C)CCO)CC(O)CN1C(=O)COCC(N1CCCC1)C 83113,Cc1cc(Cl)ccc1C(=O)NCC1CCC(C)N(C(=O)CSC(F)F)C1 83114,c1(OC)cncc(C=CC(=O)NC2CCCC2CNC(c2ccc(Cl)o2)=O)c1 83115,C12(NC(CCCSCC)=O)CCCC1N(C(c1ccc(OC3CC3)cc1)=O)CC2 83116,C12(CNC(c3c(CC)noc3C)=O)CCCC1CN(C(C1CC3(CC3)C1)=O)C2 83117,N1(C(C=C(CCC)C)=O)CCN(C(c2cc(F)cc(Cl)c2)=O)CC1C1CC1 83118,CC1(C)OCCOC1CC(=O)NC(C)(CNC(=O)C=CC=C(Cl)Cl)CO 83119,C1(CC(=O)NCC(C2CCCCC2)NC(c2c(C)coc2)=O)CCC(=O)N1C 83120,c1(C(C(N2CC(CNC(C=NOC)=O)(OC)C2)=O)O)ccc(Cl)c(Cl)c1 83121,C(C(C)C(C)C(=O)N(CCCCCNC(c1ccoc1)=O)C)OC 83122,C1(C(N2C(CNC(c3c(C)nn[nH]3)=O)CC2)=O)CC(C)CC(C)(C)C1 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83140,N1(CC=C(C)CSc2ccccc2)CCCC(O)C1C(C)C 83141,C1(NC(c2c(C)ncs2)=O)CCC2(CC1)CC2NC(c1snc2ccccc12)=O 83142,C1(CNC(C=CC)=O)CN(C(c2cncc(C(F)(F)F)n2)=O)CCO1 83143,C(c1ccc(F)cc1)=C(C(=O)NCC1(C)N(C(C=CCC)=O)CCC1)C 83144,c1(C(N2CC(NC(CC(N3CCCCC3=O)C)=O)C2)=O)cc2ccccn2c1 83145,C1(C(=O)Nc2c(C)ncnc2)CC(F)CN(S(=O)(=O)C(F)(F)F)C1 83146,c1(SC)ccc(C(=O)NC(C2CCCC2)CNC(=O)C(C)OC2CC2)s1 83147,c1(C(N2CC(N(C(CCCOCCC)=O)C)C(O)C2)=O)cccc2c(C)[nH]nc12 83148,c1(-c2scc(C(N3CCCC3c3cccs3)=O)n2)ccccc1F 83149,C=C(C)CC(C(=O)NCCOC(C)=O)NC(=O)CCO.CCCCOC 83150,Cc1ccc(C(=O)C(=O)NCCCCC(C)NC(c2cnc(Cl)cn2)=O)cc1 83151,C(=O)(C(C)CCCCCCC)N1CCN(C(C2CC(C#C)(O)C2)=O)C(C)C1 83152,N1(C(CCc2cccc(C)c2)=O)CCN(C(C2CC2F)=O)CC1C 83153,N1(C(c2c(SC)ccs2)=O)CC2C(CNC(=O)Cc3ccsc3)C2C1 83154,N1(CC(=O)N(C(C)(C)C)C(c2cnc(C)nc2)=O)CCCC(C)(N(C)C)C1 83155,N1(C(c2ccn(COC)n2)=O)CC=CC1(C)C(=O)NCc1nccc(C)n1 83156,c1(OC)cc(C(N2CCOC(C(=O)NC3CSCS(=O)(=O)C3)C2)=O)cc(OC)c1O 83157,CS(=O)c1cccc(C(=O)NCC(CO)NC(c2ccnnc2)=O)c1 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83176,CCC(C)C(C(=O)N1CC(NC(c2cnc(N3CCCC3)s2)=O)C1)OC 83177,N(C1CCc2c(Br)ccc(Cl)c21)C(C1C2(C(=O)O)CC(C)(C2)O1)=O 83178,C1(C(=O)NC2(CC=C)CCN(C(=O)Cc3cnns3)C2)CCC=CCCC1 83179,C1(C(=O)NCC#CC(=O)NC(C=C)(C)CC)CC2(CCC2)CO1 83180,c1(C(=O)NC(C2(CNC(C)=O)CC2)C)ccc(C#N)c(F)c1Br 83181,C1(NC(c2c(NC)snc2C)=O)CCC2CCN(C(c3cc(C(N)=O)c[nH]3)=O)C12 83182,C1(C(N2C(CNC(C(N3CC(C)C3)C)=O)CC(F)C2)=O)NC(=O)OC1(C)C 83183,c1(C(=O)NC2C(C)CN(C(=O)C(C)(C)C3CCOC3)C2)cn2ccsc2n1 83184,C1(C(N2C(C)CC(CNC(c3c(CC)csc3)=O)C2)=O)CC2CCC(C1)C2=O 83185,N1(C(CNC(CNC(c2n(C)ccc2)=O)=O)=O)CC2(CCC2)CC1CO 83186,O=C(N=S1(=O)c2ccccc2Nc2ccccc21)C1COCCC1(F)F 83187,C12COCCC1C(=O)N2.c1(NC(=O)CN2CC(COC(F)F)C2)cccc(O)n1 83188,C=CC1CN(c2cc(C)nc(N3CCCC(CCO)CC3)n2)CCO1 83189,N1(C(=O)Nc2cncs2)CC2CCN(C(c3coc4ccccc34)=O)C2C1 83190,C(=O)(C1=C(c2cscn2)N(CCSC)C(=O)NC1c1ccc(C(F)F)o1)OCC 83191,N1(C(CC2CN(C(CCC(=O)NC)=O)C(C)C2)=O)CC2(CCCCC2)C1 83192,CC(CC(=O)N(CC(C)NC(=O)Cc1nnc(O)s1)C)P(C)(C)=O 83193,c1(CNC23CCC(NC(C4CN(C)C4)=O)(CC2)C3)c(F)ccc(Cl)c1F 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83212,N1(C(c2cc(C)cc(Cl)c2O)=O)CCC2(CC1)CCN(C(=O)OC(C)(C)C)CC2 83213,n1(CC(=O)NC2C(CNC(CN(C)C)=O)CCC2)cccc(O)c1=O 83214,c1(C(=O)NC(CC(C)C)CNC(=O)CC#N)cccc2cccnc12 83215,CC1(C)CCc2c(C(N3CCN(C(=O)CCC(N)=O)CC(C)(C)C3)=O)csc2C1 83216,c1(CC(C)C(=O)NCCCOCCNC(C2CCC(=O)N2)=O)ccccc1F 83217,Cc1cc(C(N2CC(NC(c3cnc(Cl)cc3I)=O)C(C#N)C2)=O)cc(C)c1F 83218,Cc1cc(C)c(C(=O)N(CC(C)NC(c2ccnc(CC(C)C)n2)=O)C)cc1N 83219,C1(CCC(=O)NCC(C=C)O)CCN(C(=O)Cc2cccs2)C1 83220,CCCC(CCCNC(C1(C)CCC(=O)N1)=O)NC(=O)C(C)n1cnnn1 83221,c1(OC)c(Cl)ccc(C(=O)NCC2(O)CN(C(=O)C(C)(C)SC)C2)c1N 83222,C(=O)(C(C)(C)C(C)NC(=O)CN1CC2CCC1C2)NC(CC)C(F)(F)F 83223,c1(OC)ccc2c(c1)C(C(=O)N(CCCNC(=O)C1=CS(=O)CCC1)C)CCC2 83224,c1(C(N2C(C)CC(CNC(CCCCC)=O)C2)=O)ncc(Cl)c(N)c1Cl 83225,N1(C(CCN(C)CC)=O)CCN(CC(=O)NCc2ncc[nH]c2=O)CC1 83226,C1(NC(=O)C2=CCC2)CC2(CCC(NC(C3CC4C=CC3CC4)=O)CC2)C1 83227,c1(C(=O)NC2C(NC(C3N(C(C)=O)CCC3)=O)C2)c(Cl)cccc1Cl 83228,Cc1cccn2cc(CC(N3CCN(CCNC(=O)C(C)C)CC3)=O)nc12 83229,N1(C(CC(C)F)=O)CC2CCC(CNC(=O)C(C3CC3)C3CC3)C2C1 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83247,C1(C(=O)NCCC(=C)CNC(c2cc(C)n(C)n2)=O)CCOC(C)(C)C1 83248,C1(CNC(COC)=O)CCCC1C(=O)NCc1csnc1C 83249,c1(N(C(C2CCCNC2)C)Cc2ccc(Br)c(F)c2)ncnc2cc(I)sc12 83250,C1(F)(C(N2CC(NC(COCCCC)=O)C(C(F)(F)F)C2)=O)CCS(=O)(=O)C1 83251,C(=O)(CC(CSC)NC(=O)CC#N)NC(C#C)CC1CCC1 83252,c1(C(N2CCCCC2CCN(C)C)C(=O)NC(CC)C)nccnc1OC 83253,N1(C(C)=O)CCN(C(=O)CCC(=O)c2ccc(F)cc2)CC1.C(C(=O)C1(Cl)CC1)NC 83254,C1(C)(Cn2cc(-c3ccc(C(=O)NC(C4(CO)CC4)C)cc3)nn2)CCC(=O)N1 83255,C1(CC=C)(NC(=O)C=Cc2ccncc2C)CCCN(C(C2(C)CC2Br)=O)C1 83256,C1(O)(C(C)NC(=O)CCOc2cccnc2)CCN(C(=O)C=CC2CC2)CC1 83257,c1(NC(C2N(C(C(CSC)OC)=O)CCC2)=O)cnc(Cl)nc1 83258,Cc1nnc(CCC(=O)NC23CC(NC(=O)CCN4CCC(O)CC4)(C2)C3)n1C 83259,C1(C(N2CCC(c3cn(-c4ccccc4)nn3)C2)=O)CCS(=O)(=O)C2(CCC2)C1 83260,C1(NC(C=CC(C)C)=O)C(CNC(C2(S(C)(=O)=O)CCCC2)=O)CCC12CCC2 83261,C=CC(C)(CC)C(=O)NC1CCC(CN(C(=O)C(c2ccc(Cl)cc2)=O)C)CC1 83262,Cc1c(CNC(=O)C(C[Si](C)(C)C)NC(=O)OC(C)(C)C)cnc(Cl)c1Br 83263,N1(C(C=CCCC)=O)CCC(CNC(=O)C(C)Oc2cccc(CO)c2)C12CC2 83264,CC1CCCC1(C)C(=O)NC1CCC(NC(C2(Cc3cnn[nH]3)CCC2)=O)CC1 83265,c1(OC)cccc(Cl)c1C(=O)NC(C)CC(C)NC(c1cnoc1C1CC1)=O 83266,C1(CN2C(C)C(C(=O)O)CC2)CCC2C(C1)C2(F)F 83267,c1(C(CC)C(=O)N(CCNC(=O)C=CC(C)C)C(C)C)ccc(OC)cc1 83268,c1(C(=O)NC2CC(n3cc(-c4cscn4)nn3)C2)ccc2c(c1)CCO2 83269,C(CCCCC(=O)NCC(O)C(F)(F)F)NC(c1c(C)cncn1)=O 83270,N1(C(c2cc(COC)[nH]n2)=O)CCOCC(C(N2CCSC(C(C)C)C2)=O)C1 83271,C(CC(C)C)(C(=O)NCC(c1ccccc1)NC(c1ccn(CC#N)n1)=O)OC 83272,C(=O)(C(CNC(C1(O)CCOC1)=O)C(C)(C)C)NCCC(CC)(C)C 83273,c1(NC(=O)CC2CC(NC(=O)CC3CC(C(=O)NC(C)(C)C)C3)C2)n[nH]cc1Br 83274,CCC(O)CC(=O)NCC1(NC(=O)Cc2cncc(C)c2)CCOC1 83275,C1(C(N(C(C(=O)OC)C)C)=O)(NC(C2CC2(F)F)=O)CCN(C)C1 83276,c1(C(=O)NC2C(NC(CCc3c(C)cccc3)=O)CCCC2)ncc(F)cc1F 83277,C1(C(=O)NC)CCCN(C(=O)CC2(C)CCN(C(c3nccnc3OC)=O)C2)C1 83278,c1(C(C(=O)NCC(C)(CO)NC(c2cn(C)nn2)=O)O)ccc(Br)cc1 83279,c1(CCNC(CN(C(C)C)C)=O)ocnc1CNC1CCCC1.C(=O)CC1CC1C 83280,N(C(=NCCN1CCCC1)NCC1CCOC1)CC(C)(C)CSc1ccccc1 83281,N(C(=NCCCCc1cn[nH]c1)N1CCC(C2CCOC2)C1)CC(O)C(F)(F)F 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83299,N1(C(CCC(=O)N(C)C)=O)CCCC2(NC(c3nncn3C)=O)CC2C1 83300,c1(NCC(O)CC2CCCO2)ccc2nc(Cl)ccc2c1 83301,c1(-c2nn(-c3cnccc3)c(C3CC4(C3)CC(F)(F)C4)n2)cccc2ccsc12 83302,c1(C(=O)NCc2cn(CCNC(c3ccn(C)n3)=O)nn2)[nH]cnc1C#N 83303,C1(C(=O)NCC(CNC(c2cccc(F)c2)=O)O)CC2(C1)CC2(F)F 83304,c1(SC)nc2ncnc(N3CCCC(CCNC(=O)COC4CCOC4)C3)c2s1 83305,c1(C(N2CC(CNC(c3cc(C)[nH]c3C)=O)C3(C2)CC3)=O)ccnc2c1CCO2 83306,c1(C(=O)NC(C2CCN(C(c3cccc(NC(C)C)c3)=O)C2)C)cc(Cl)nnc1O 83307,C=C=C(C)CC(=O)N(C1CCN(C(=O)CNC(=O)C2CC2)C1)CC 83308,C1(C)(CNC(c2cc(CC)on2)=O)CCC(NC(=O)C=Cc2ccnn2CC)C1 83309,CC(C)(CNC(=O)CCCn1ccnc1)CC(=O)NC(C1CCOC1)CO 83310,c1(C(N2CCC3CCC(C2)S3=O)C(=O)NC2CCC2)csc2ccccc2c1=O 83311,c1(C(C(=O)NC)N(C)CC2CCCO2)cc(Br)c(F)cc1F 83312,C=CC1(O)CCN(C(=O)CNC(=O)CNC(c2nn(C)cc2C)=O)C1 83313,c1(C(N2C(CCC)COCC2)C(=O)NCCC)ccc(C)c(C#N)c1 83314,N1(C(c2cc(F)ccc2Br)=O)CCC2C1CCN2C(c1ccsc1)=O 83315,Cn1cc(C(N2CC=CC2(C)C(N2CCCCC2CC(N)=O)=O)=O)ncc1=O 83316,c1(C(N2CCCC(NC(C(C)c3cccs3)=O)C2C)=O)ccc(F)c(F)c1F 83317,c1(C(=O)Nc2scc(-c3ccc(OC)cc3OC)c2)cc(Cl)c(Cl)cc1Cl 83318,N1(C(CC2C(C)=NNC2=O)=O)CC2CC(C1)C2NC(=O)CCC(C)(C)C 83319,c1(C(N2CC3C(CNC(=O)C=CC4CCOC4)(C3)C2)=O)cc2c(nn1)CCOC2 83320,C(CC(F)F)(C(=O)N(C)CCC1CCCC1)NC(C1C(OC(C)=O)C1)=O 83321,c1(C(N2CCCC(CCNC(c3c(COC)ncs3)=O)C2)=O)ccc(C)c(O)n1 83322,C1(NC(C2CN(C(=O)CCC3CCCCO3)CC2F)=O)CCCC(O)CC1 83323,Cc1ccc(CN(C(=O)CCOCCCNC(=O)Cc2conc2C)C)cn1 83324,c1(C(=O)OCC)ccc(NC(=O)N(C2CC3(C2)CC3F)CCN(C)C)cc1 83325,C=CCC(CNC(=O)CC1CCCCCC1)C(=O)N(CCCOC(C)C)C 83326,c1(C(=O)NCc2cccc(C#C)c2)cc(F)c(F)cc1F 83327,c1(CC(=O)NC2CC3CC2N(C(=O)CC2NC(=O)NC2=O)C3)ncc(F)cc1F 83328,C1(OC)(CNC(=O)CN=[N+]=[N-])CN(C(=O)CCSC)C1 83329,c1(C(N2CC(C3(NC(=O)Cc4ccc(Cl)s4)CC3)C2)=O)cc2c(=O)[nH]ccn2c1 83330,C1(NC(C2(C)CCOCC2)=O)CC(CO)C(O)C1O.C12CN(C1)C(=O)CO2 83331,C(CCN=C(NCC(N1CCOCC1)C)NCC1(O)CCC(C)(C)CC1)SC 83332,C1(C(=O)NC(CNC(=O)C(C2CC2)C2CC2)C2CCC2)CC12CCCC2 83333,Cc1ccc(C(=O)NC2CCN(C(c3ccc(CN(C)C)o3)=O)CC2C)c(O)n1 83334,c1(C(N2CCN(C(c3cnc(C(C)C)s3)=O)CC2C)=O)cnc2c(c1)CCCO2 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83352,Cn1cc(CCC(=O)NCC2CCC(NC(=O)CC3CCCOC3)C2)cn1 83353,c1(NC(C2CCN(c3c(Cl)cnc(C)n3)CC2)=O)ncc(C#N)cc1I 83354,c1(CC)c(C(=O)NC(C2CCN(C(=O)CCCCSC)C2)(C)C)cnn1C 83355,C(CCC(C)C(=O)NCC(C)(C)CCNC(c1sccc1OC)=O)OC 83356,N1(C(c2nc(COC)sc2)=O)CCC2(CCCC2NC(c2[nH]c(C)nc2C)=O)C1 83357,C#CCCCCC(=O)NC(C)(CNC(c1cn(C2CCOC2)cn1)=O)C1CCC1 83358,C1(C(=O)NC(CNC(CC(=O)OC)=O)(C)C2CCC2)CCCC12CCOCC2 83359,C1(NC(CC2N(CC)CCC2)=O)CN(C(c2cc(O)cs2)=O)CC1C(F)(F)F 83360,C(CC1CCC1)(C(=O)N1CCCC1CC(N)=O)NC(C(C)=C(CC)C)=O 83361,C1(C(=O)NCC2=C(C)CCC2)CC2CCC(C1)N2C(c1c[nH][nH]c1=N)=O 83362,Cc1oc(C(=O)NC2CCN(C(=O)CCc3cccc(O)c3)C2C)cc1Br 83363,C1(CC)CC(O)CN1C(=O)CC1CC(NC(=O)CC2OCCC2C)C1 83364,C(=O)(C(C)C(=O)NCC1(CC(=O)NC(c2cncs2)C)CC1)OC 83365,N1(C(CC)=O)CC2(CCCC(CNC(c3ccc(C)c(S(N)(=O)=O)c3)=O)O2)C1 83366,C1(C(F)F)(NC(CC(C)(C)CNC(=O)CC2CC23CC3)=O)CCCCC1 83367,c1(OC)cc(C(N2CC(F)CC2CN(C(=O)C(c2cnn(C)c2)C)C)=O)n(C)n1 83368,c1(C(=O)NCC2=CCN(C(=O)Cc3ccccc3F)CC2)cc(Cl)ncc1F 83369,c1(CCC(=O)NCC(CCNC(C)=O)F)ccccc1-n1cc(CO)nn1 83370,C(=O)(CC1=NN(C)C(=O)C1)NC(c1nocc1C(=O)NCC1(C)CCC1)C 83371,c1(C(=O)NC2CN(C(CC(CC)SC)=O)CC(O)C2)cncc2sccc12 83372,c1(NC(c2n(C(C(=O)OC)C)nnn2)(C2CC=CC2)C)cc(C)cc(Br)c1 83373,c1(C(=O)NCC(c2ccccc2)NC(C(C)SCC)=O)cccc(F)c1C 83374,CC(C)CC(C(=O)N1CCCC1CCNC(=O)CC1CCC(=O)NC1=O)N(C)C 83375,C1(CNC(C(CCC)(C)CCC)=O)CC2(CCOCC2)CN1C(c1csnn1)=O 83376,N1(C(C=C(C)C)=O)CC2CC(NC(c3cc(C)on3)=O)C2C1 83377,C12(C(=O)NCCCN(CCCNC(C)=O)C)CCC(C1)c1ccccc12 83378,N1(C(C2CCC(=O)N2)=O)CC2CC(NC(c3cc(C(F)F)[nH]n3)=O)C2C1 83379,c1(C(=O)NC(CCOC)CNC(=O)C(O)c2ccco2)ccc(C2CCC2)nc1 83380,N1(C(CCS(C)(=O)=O)=O)CCC(NC(C2CC(C)(F)C2)=O)C(F)(F)CC1 83381,C1(N2C(=O)CN(CC3CC3)C2=O)CN(N2CCN3C(=O)NCCC3C2)C1 83382,Cn1c(C(=O)NCC2COC(CNC(=O)CCCCCF)C2)cc2occc12 83383,CN=c1[nH]c(=NCc2cc3c(s2)CCCC3)[nH]c(=NC(C)c2ccc(Cl)cc2)[nH]1 83384,c1(CC)nn(C)cc1C(C)NC(=O)Nc1cccc(OC2CC2)c1 83385,c1(C(=O)NCC(CNC(C(C)n2cnnn2)=O)F)c(F)cccc1Br 83386,C1(C(N2C(C3(C(=O)NC(c4ccc(O)cc4)C)CC3)CCC2)=O)CC1C1CCC1 83387,C1(O)(CN(C)C(C2CCC(F)(F)C2)=O)CCCN(C(c2ccc(C3CC3)o2)=O)C1 83388,C1(NC(C(CC)c2ccccc2)=O)CC(F)(F)CC1NC(c1ccc(Cl)cc1)=O 83389,c1(CN(C2CCC23CCNCC3)C(C2CCCCO2)=O)cccc([N+](=O)[O-])c1F 83390,C1(C(N2CC(CCNC(C3CS(=O)(=O)C3)=O)OCCC2)=O)CCCC2(CCC2)C1 83391,C(=O)(CC(C(=O)NC1CC(NC(c2coc(Cl)c2)=O)C1)N1CCC1)OC 83392,S(=O)(=O)(c1ccc(Br)cn1)N(C1CCNCCC1C)c1ccc(SC)cc1 83393,C1(C(=O)NCCc2c(C(=O)NC(CC)C(C)(C)O)c[nH]n2)CCCCC(=O)C1 83394,CCCC(CCCNC(=O)C(O)CF)NC(=O)CN(C1CCC1)C 83395,C#CCCCC(C)C(=O)NC1CC12CCN(C(c1ccccc1C(C)=O)=O)CC2 83396,CC1(C)CC(C)(C(=O)NCCCC(F)(F)F)CN1C(C1CCC(=O)NC1)=O 83397,Cc1ccc2c(C(=O)NC3C4CCC(C4)C3C(=O)O)n[nH]c2c1 83398,C1(NC(c2c(C)csc2)=O)CCCCC12CCN(C(=O)C(C)(C)C(F)(F)F)C2 83399,C1(C2CCN(C(c3cn(C(C)(C)C)nn3)=O)C2)(NC(C2=C(C)CCC2)=O)CC1 83400,C1(CNC(C2(CCOC)CC2)=O)C2CCC(C2)N1C(c1ccc(Cl)cc1F)=O 83401,C1(C(N(CCC(C(C)C)NC(c2nc(=O)n(C)[nH]2)=O)C)=O)CCS(=O)(=O)C1(C)C 83402,C1(NC(c2c(OC)n(C)nc2)=O)COC2C(NC(=O)C(C)C(=O)C3CC3)COC12 83403,CCC(CN(C)C)CC(=O)NCC1CCN(C(c2cc(COC)on2)=O)CC1O 83404,c1(CC(=O)NCc2scc(CNC(C=COCC)=O)n2)cc(O)nc(O)n1 83405,N1(C(CC(C=C)(C)O)=O)CCN(C(=O)C(C2CCOCC2)O)C2(CCC2)C1 83406,CC(C(=O)NC(C)Cn1cc(-c2cc[nH]c(=N)c2)nn1)C(F)(F)C(F)F 83407,c1(OC)ncc(C(=O)NCC2CC(NC(C3(OC)CC3)=O)CC2O)cc1Br 83408,c12cc(cs1)COC2=O.C(CCC(C)=C(C)CCC=CCON)=C(C)C 83409,CCCCC(C(=O)NC)NC(C12CC(CO)(CN1C(C1(CC)CCCO1)=O)C2)=O 83410,Cc1c[nH]nc1C(=O)NC(CNC(C1(C)CC1(Cl)Cl)=O)CO 83411,Cc1ccc(CC(=O)NC(C2COCCN2)C)cn1 83412,c1(OC)ccc(C(=O)N(C2CCN(C(=O)C3=NOC(C)C3)CC2)CCO)c(Cl)n1 83413,C1(CC(=O)N(CCCCNC(=O)CCN2CCCC2)C)CCC2CC12 83414,Cc1[nH]nc2c1CCN(c1nnc(C3CCS(=O)(=O)C3)n1CCC(=O)N(C)C)C2 83415,c1(COCC)cc(OCc2cccc(OCC)c2)c(C(=O)NC2CCCO2)[nH]1 83416,c1(CC(=O)NCC(C)N(C(CCCOCCOCC)=O)C)cccc(F)c1F 83417,c1(N(C(=O)C(C)C)CCNC(c2ccc(N(CC)CC)cc2)=O)ccc(C#N)cc1 83418,C(C)(CC(C)NC(C1(CC(=O)NCC2CCCC2)CCCC1)=O)NC(CCC)=O 83419,c1(C(=O)OC)cnc(OC)c(C(N2CCC(NC(c3ccccc3)=O)C2C)=O)c1 83420,c1(C(N2CC(NC(C(CCC#C)O)=O)CC2(C)C)=O)cc(N)c2ncccc2c1 83421,c1(OCC)ncc(C(=O)N(CC(C)NC(=O)C(O)CF)C)s1 83422,CC1(C(=O)NCC2(F)CC(CNC(=O)C3CC3)C2)CC(C(F)(F)F)=NO1 83423,C(C(C)C(=O)NNC(=O)Cc1ccccc1[N+](=O)[O-])SC 83424,N1(C(C(=O)Nc2cccc(C(=O)OCC)c2)C2CC2Cl)CCn2ncnc2C1 83425,C[S+](C)CCC(O)C(=O)N1CC2CCC2(CNC(c2cccc3nc[nH]c23)=O)C1 83426,C1(C(N(C2CC3CCC2O3)C)=O)C(O)CCN1C(=O)C(=C1CCCCC1)F 83427,C(c1ccccn1)=C(C)C(=O)NC(C(F)(F)F)c1ccc[nH]1 83428,c1(C(C)C)nocc1C(=O)NCC(C)(CO)NC(=O)COC1CCOC1 83429,Cc1ccc(SCC(N2CCN(c3cc(-c4cc(N)ccn4)ccn3)CC2)=O)cc1 83430,C(CC(C)(C)CC(=O)NCC1CC(NC(c2nc(C)n(C3CC3)c2C)=O)C1)OC 83431,CC(O)C(C(=O)NCC(c1ccccc1)NC(c1coc(Cl)c1)=O)N(C)C 83432,C1(NC(C23N(C(c4ccc(Cl)cn4)=O)CC(C2)C3)=O)CCCCCC1F 83433,c1(C(N2CC(O)(CCNC(C(COC)OC)=O)C2)=O)nn(C)cc1S(C)(=O)=O 83434,C1(NC(C=CC(=O)OCC)=O)CN(C(=O)CC(C)C2CCCCC2)C2CCCC12 83435,C#CC1(C(=O)N(C)CC2CC2C)CCN(C(C2CC(C)CCO2)=O)CC1 83436,C12(NC(CCCCC)=O)CCCCCC1N(C(=O)CC(C)(C)CC(=O)OC)CC2 83437,C(=O)(C(C)(CC)NC(=O)NC(C(=O)NC)CCSC)OC(C)(C)C 83438,CC1(C)CC(C(N2CCn3ccnc32)=O)CN(C(=O)C=Cc2cscn2)C1 83439,Cc1cc(C(=O)NCC(O)CNC(C2CC(C)(C)CO2)=O)c(C)o1 83440,N1(C(CC(CN(C)C)OC)=O)CCC(O)C(C)(O)C1.C1(C(=O)N)(CO)CCCC1 83441,c1(N2CCC(CNC(C(C3CC3)OC)=O)C(C)C2)ncnc2c1CCC2 83442,CCCCC(C(=O)NCCCCC(=O)NC(c1cncn1C)CO)N(C)C 83443,n1(CC(=O)NC(CNC(CC)=O)(CC)CC)ccc2ccc(Br)cc12 83444,CN1C(C(=O)NC2(C(=O)NCc3ccc(O)cc3F)CC2)CCS1(=O)=O 83445,N1(C(c2n(CC)ncc2Br)=O)CC(NC(=O)C(C)CF)C(S(C)(=O)=O)C1 83446,c1(C(=O)NC2CCN(C(Cc3c(C)noc3)=O)CC2F)cn2ncccc2n1 83447,c1(OC)ccc(CC(=O)N(C(C)CNC(C2CCCOC2C)=O)C)nc1 83448,N1(C(c2cncn(C)c2=O)=O)CC2CN(C(=O)C(CO)NC(N)=O)CCC12 83449,c1(C(=O)NCC(c2ccc(C)cc2)NC(C2CCC3CC23)=O)ccc(C)c(C)n1 83450,Cc1ccc2nc(C(=O)NC3CCCC(NC(=O)CC(C)N(C)C)C3)cn2c1 83451,N1(CC(=O)NCCCC2(NC(C(C)OCC(C)C)=O)CC2)CCCS1(=O)=O 83452,C12(C(=O)NC(C(C)C)CNC(C3CC3c3ccccc3)=O)CCC(CC1)O2 83453,C(=O)(C1=C2CCN=C2NC=C1)N1CCC2(OCC(NC(c3c(C)nco3)=O)C2)C1 83454,CN1CCC(=CC(=O)NCC2CCC2NC(=O)CNC(=O)CC2CCCC2)CC1 83455,N1(C(COCC)=O)CC(F)(F)CC1C(=O)NCC1(O)CCCOC1 83456,c1(OC)ccc(C(=O)N(CC(C)(C)NC(=O)C(C)Cn2ccc(C)n2)C)c(F)n1 83457,Cc1oc(Cl)nc1C(=O)NC(C1CCN(C(=O)CCc2cn(C)nn2)C1)C 83458,C=CCC(Cc1ccccc1)C(=O)OCCCCOCCCO 83459,C1(C(=O)NC(c2occ(C(N(CC(=C)C)CC)=O)n2)C)C2CC3C(C2)C13 83460,N1(C(C(C)(F)F)=O)CC2(CCN(C(C3CCCC4(CC4)C3)=O)CC2)C1 83461,c1(C(N2CCCC(NC(C(CC)CC)=O)C2C)=O)cc[nH]c2nccc1-2 83462,C1(NC(Cc2cc(C)no2)=O)CCCC12CCN(C(=O)C(O)c1ccsc1)CC2 83463,C#Cc1ccc(C(N2CCCC(C)(NC(=O)Cc3nnc(O)s3)C2)=O)cn1 83464,c1(NCC(=O)NC(C)(CNC(=O)CC2NC(=O)NC2=O)CO)ccc(F)cc1F 83465,C1(C(=O)NC(C(=O)NC(c2ccncc2F)C)C2CC2)CCCC(O)C1 83466,N1(C(c2[nH]ccc(=N)n2)=O)CCC2CCN(C(c3cc(C(F)F)no3)=O)CC2C1 83467,N1(C(C)=O)CC=CC1CNC(=O)Cc1cc(C(=O)NC(C)(C)C)on1 83468,c1(C(N2CCCC(N(C)C(C)=O)C2)C(=O)NC)cnc(C)n1C 83469,Cn1nc(C(N2CC(c3ccccc3C(F)(F)F)(O)C2)=O)cc1C1CC1 83470,C1(CNC(c2cc(OC)no2)=O)CC(NC(=O)CCCC#N)C12CCC2 83471,N1(C(CS(=O)(=O)NC)=O)CC2(CCCC2NC(=O)CC2CC3CC3C2)C1 83472,c1(OC)ccc2c(c1)OCCC2NC(=O)NC1CCN(c2ccc(C)cc2)CC1 83473,c1(C(=O)NCCC(C)N(C)C(C2CC2c2ccc(Cl)cc2)=O)nc(Cl)ccc1N 83474,C(=O)(CS(=O)(=O)CC)N.CCS(=O)(=O)N1CC(C(CN2CCCC2)=O)C1 83475,N1(C(COC2(C)CCC2)=O)CCOC(CCNC(c2cc(F)c[nH]2)=O)C1 83476,c1(OC)cnc(Cl)nc1NC(C1(F)CCN(C(c2cc(C(C)C)nn2C)=O)C1)=O 83477,c1(C(N2CC(CC(C)NC(c3cscn3)=O)C2)=O)nc2c(cc1Cl)OCCO2 83478,C12(C(N3C(CNC(C4CC(=C)C4)=O)C(C)(C)CC3)=O)C3CCC(CC13)C2(F)F 83479,N1(C(C(F)OC)=O)CCC(NC(c2ccn(-c3ccncc3)n2)=O)C(O)C1 83480,c1(C(=O)NCC2(C)CCN(C(Cc3nnc(C)s3)=O)C2)ccn2c1CSCC2 83481,C(CS(=O)(=O)NC1(C(F)F)CCC1)(C1CCOC1)OC 83482,c1(C(=O)NCC(C)N(C(=O)Cc2nc[nH]n2)C)ccc2nnn(C)c2c1 83483,N#CC1CN(C(C2(O)CCN(C(c3cccc(C(N)=O)c3)=O)C2)=O)CCO1 83484,N1(C(c2scc(C(C)=O)c2)=O)CCN(C(=O)C(C)(C)N2CCCC2)CC1C1CCC1 83485,c1(C(CNC(C2CC2C2CC2)=O)NC(COCC)=O)cccc(Cl)c1 83486,c1(OC)nccc(C(=O)NCC2C=CCN2C(=O)C(N2C(=O)CCC2=O)C)c1F 83487,C(C(CNC(=O)CCCCC1CC1)S(C)(=O)=O)NC(c1cc(C)no1)=O 83488,c1(OC)ccnc(C(=O)NC(C)CN(C(=O)C(O)C2CC2)C)c1F 83489,C1(C(=O)Nn2cc(-c3nc(C4CCCO4)no3)nn2)CCCC1C(F)F 83490,C(CNC(=O)C(C)n1ccnc1)(CC(=O)NCC(C)C(C)O)OC 83491,c1(C(N(CCN(C(C2C(CC)CCC2)=O)C)C(C)C)=O)cc(=O)n2nccc2[nH]1 83492,CC(C)(C(=O)N1CCC(CCO)C1)C1=CCN(C(c2ncccc2Cl)=O)C1 83493,CC1(C(=O)NOCC2CCCO2)CCN(C(C2CC23CC3)=O)CC1 83494,C(=O)(CCS(C)(=O)=O)NCC1OCC(CNC(c2c(OCC)cccc2)=O)C1 83495,C(C1=NOC2CCCC12)NC(C1(F)CN(C(C2CC(=C)C2)=O)C1)=O 83496,CC(C)CS(=O)(=O)CC(=O)NC1CC2(C1)CC2NC(=O)CN(C)C1CC1 83497,N1(C(CCSCC)=O)CCN(C(=O)CCc2ccc(OC)cc2)C(CC)C1 83498,C1(NC(C2(C(N(C(C)C)C)=O)CC2)=O)CCCC1NC(=O)C1=CCC1 83499,c1(C(=O)NC)cccc(OC(C)C(=O)NC(C)CNC(c2c(C)coc2C)=O)c1 83500,CC1(C)C(C)(C)C1(F)C(=O)NC1CN(C(c2c[nH]ccc2=N)=O)C2CC12 83501,C1(C(N2CC(O)(CNC(c3cn(C4CC4)cn3)=O)C2)=O)(COC)CC1(F)F 83502,C1(O)(C(N2C(C)(CNC(=O)CSCC3CCCO3)CCC2)=O)CN2CCC1CC2 83503,C1(NC(c2cn(CC)nc2C(C)C)=O)CCCCN(C(C2CC23CCCC3)=O)C1 83504,C=C1CC2(C1)CC(C(=O)N(C1CC3CC1N(C(=O)CC1CC(C)(C)CO1)C3)C)C2 83505,C1(N(C(Cc2c(C)con2)=O)CCF)CCCN(C(C2OCC2(C)C)=O)C1 83506,c1(CC(=O)NCC(C(C)C)NC(=O)C(C)CO)cnc2n1CCCC2C 83507,C1(C(=O)OC)CN(C(=O)C(c2cccc(Cl)c2)N(C)C)CC1c1cccc(Br)c1 83508,C1(SCC(=O)N(C(C)CCNC(=O)CSC(F)(F)F)C)CCOC1=O 83509,c1(NC(N2CC(F)CC2C(=O)O)=O)cnncc1Br 83510,C1(NC(c2ccc(SC)s2)=O)CCCCN(C(C2CC3(CCO3)C2)=O)C1 83511,C1(NC(C2C(C)CCO2)=O)CC(F)CN(C(=O)CCNS(=O)(=O)C(F)(F)F)C1 83512,c1(C(N2CC3CC3(C(=O)Nc3c[nH]nc3Cl)C2)=O)cccc(I)c1Cl 83513,C1(C(N2CCC3(CC3)C2)=O)CNCCNC1 83514,c1(CC(=O)NCCN(CCOCCO)C(=O)C2CC2)ccsc1Br 83515,C(=O)(C(C)(F)C(=O)N1CC(CC(C)NC(c2ncccc2COC)=O)C1)OCC 83516,CC(C)CC(C(=O)NC(C)C(C)C(=O)N1C(CO)CC1CO)N(C)C 83517,N1(C(COCC=C)=O)CCC(C2CCN(C(c3cc(CSCC)on3)=O)CC2)C1 83518,CC1CNc2ccc(C(=O)NCCCOCCNC(C3CCCCO3)=O)cc21 83519,c1(CCC(N2CCC(Cn3cc(CC(C(C)C)O)nn3)C2)=O)ccc(F)cc1F 83520,C(=O)(C(F)C(C)CNC(=O)CCN1CCCC1=O)NCC(CC)CC 83521,C1(COCC)CCCN1C(C1CCC(n2cc(C(C)(C)CC)nn2)C1)=O 83522,c1(OC)cccc2c(C(=O)N(C3CN(C(c4n[nH]cc4OC)=O)C3)C)c(C)[nH]c12 83523,CC1CC(CNC(c2cncn2C)=O)CN1C(c1cc(C2CCC2)nn1C)=O 83524,c1(C(=O)NCCC2(NC(CC(CCC)(C)C)=O)CC2)ncc(F)c2ccccc12 83525,CC1(CC(F)(F)F)CN(NC2CC(Nc3cn(Cc4ccccc4)cn3)C2)C1 83526,Cc1cc(Br)cc(C)c1CN1CCN(C(c2cc(O)n(C)n2)=O)C(C(F)(F)F)C1 83527,N1(c2ncn(C)c(=O)c2Br)CCCC(C2CC2NC(C2(F)CC2)=O)C1 83528,N1(C(C(CNC(c2c(CC)ncnc2)=O)O)=O)CCN2CCCCC1C2 83529,c1(C(N(C2CC(NC(C3(CC#C)CCCC3)=O)C2)C)=O)ccccc1C1CCC1 83530,C1(C(N(C(CCC)C)CC)=O)CN(C(c2cnn(CCC)c2)=O)CC12CCC2 83531,c1(OC)ccc(CC(=O)NC(C)C(CO)NC(C)C)cc1[N+](=O)[O-] 83532,C1(C(N(C)CC2N(C(c3ccc(CC)cn3)=O)CCOC2)=O)CC(C)(C)CCO1 83533,C#CCCCC(C)C(=O)NC1(CNC(c2nocc2Cl)=O)CCCCCC1 83534,N1(C(C(C(=O)OCC)C2CC2)=O)CCOC2(C1)CN(C(C1CCCCO1)=O)C2 83535,C#CC1CCC(C(=O)NC2CC(C)CN(C(=O)CSc3c(C)n[nH]c3C)C2)CC1 83536,C1(NC(=O)CC2C3COCC23)CCC12CCCCC2 83537,CC(CC(=O)NC1CN(C(=O)C2=CCC2)CC1N(C)C)C(=O)c1ccc(Cl)cc1 83538,CC1(CNC(C2(F)CN(C(=O)Cc3cscn3)C2)=O)NC(=O)NC1=O 83539,c1(C(=O)NCCn2cc(C(N(C)Cc3nnc(O)o3)=O)nc2)cccnc1S 83540,N1(C(c2ncc(CC)cn2)=O)CCC(CO)(CNC(c2cnsn2)=O)CC1 83541,CCC(CCc1ccccc1)NC(c1ncc(I)s1)CC 83542,C#CC1CN(C(=O)CS(=O)(=O)CCC)CCN1C(=O)CC(C)P(C)(C)=O 83543,C1(CCCCNC(CCOCC)=O)CCN(C(=O)C(O)CC2CCOCC2)CC1 83544,C#CCC(CC(F)F)C(=O)N(C1CCC(NC(=O)C2=C(Cl)CCC2)CC1)C 83545,c1(SC)cc(C(=O)N(CCCNC(=O)CCCn2cccn2)C2CC2)nn1C 83546,Cc1c(CCC(=O)NC(C)CC2CN(C(=O)C(CCO)N(C)C)C2)cnn1C 83547,c1(C(=O)NC2CN(C(CCCCC#C)=O)CC(O)C2)cncc2n[nH]cc12 83548,C1(C(=O)NC(c2ccc(F)cc2F)C)C2CCC(C2)C1N 83549,c1(CC(=O)N(CC(C)(C)NC(C(C)O)=O)C)cnnn1C 83550,c1(NC2CCN(CCOC)C2)cc(Br)ccc1S(=O)(=O)NCc1ccc(Cl)nc1 83551,CCC(CC(=O)NCc1cccnc1NC(C1(COC(C)C)CC1)=O)SC 83552,C1(C(=O)NCCN(C(C2CCCC23CCC3)=O)CC)CN(C)CC(C)O1 83553,c1(C(N2CCC(C)(NC(=O)Cc3ccns3)CC2)=O)ccc2sccc2c1 83554,c1(C(=O)NCC(CC)(C)NC(C2(C)CCCCO2)=O)cc(C2CC2)nn1C(C)C 83555,CC1CCCCN1C(C1(CNC(=O)C(C)OC2CCCC2)CC=CC1)=O 83556,Cn1cccc(C(N2CCC3C(C(=O)OC(C)(C)C)C3C2)=O)c1=O 83557,C(C(CC1CC1)C(=O)NCC1C2CCCCC12)NC(c1ccc(CC)o1)=O 83558,c1(C(=O)NC2C(CNC(Cn3nnc(=N)[nH]3)=O)CCC2)cccn2nccc12 83559,CC1CCN(C(C23CCCN2CCC3)=O)CCN1C(=O)C(F)(F)c1nccn1C 83560,CCCC(CNC(C1CCCCCN1C)=O)C(=O)NC1CCCCC1CCO 83561,N=c1[nH]cc2c(c1C(N1CC3(CCN3C(C3C=CCC3)=O)C1)=O)CCC2 83562,N1(C(CCCC(C)O)=O)CCCC12CCN(C(c1cc(Cl)c(Cl)[nH]1)=O)C2 83563,C1(C(=O)NC2(C)C(C)CCC2)C2CCC(C2)N1C(c1ccc(F)s1)=O 83564,C12(C(=O)NC)CCCCC(=O)N1CCC2.c1(NC(C)=O)nc(CN(C)C2CC2)cs1 83565,CCCCCC(C)(C)C(=O)NCC(O)CNC(c1nnn(CC)c1C)=O 83566,c1(C(=O)NC2C3CN(C(c4cc(C)c(C)nn4)=O)CC32)cccc2nsnc12 83567,N1(C(C2CCN(CC)C2)=O)CCCC2(CCCN2C(C23CC4CC2C3C4)=O)C1 83568,c1(C(=O)NCCCCC#C)ccc2c(c1)C(=O)N(C)C2=O 83569,C=CCCCC=CC(=O)NCC=CCNC(C1(CO)CCCO1)=O 83570,C12(NC(c3cnn(C)n3)=O)CCOCC1CN(C(=O)Cc1csc(C3CC3)n1)C2 83571,c12ccc-1cc2.c1(C(=O)NCC(O)CO)cc(-c2ccc(O)cc2)ccn1 83572,N1(C(C(CC=CC)C)=O)CCc2cc(CNC(c3cccs3)=O)ccc2C1 83573,c1(CNC(CC=C)=O)cc(C(=O)NC(C)C(C)COC)n[nH]1 83574,c1(C(=O)NC2(CNC(C3COCC(C)O3)=O)CCCCC2)cccc2ccoc12 83575,N1(C(C2C(C(C)C)OCC2)=O)CCOCC(C(=O)NCC2CC3(CCO2)CC3)C1 83576,C(=O)(CCCCC(C)(C)C)N(c1ccc(NC(=O)C(=O)NCC2CC2)nc1C)CC 83577,CN1C(=O)C(NC(c2cccc(C#N)c2Cl)=O)c2cc(Br)ccc21 83578,N1(CC(=O)NC(C2(O)CCN(C(C3(C=C)CC3)=O)C2)C)OC(C)(C)CC1=O 83579,C(=O)(CC(C)C(=O)NCC=CCNC(=O)C=Cc1ccc(OC(F)F)cc1)OC 83580,N1(C(C(C)C(F)F)=O)CCN(C(C2(C#N)CCSCC2)=O)CC1CF 83581,N1(C(C2C3CN(C(C4N(C)CC(O)CC4)=O)CC32)=O)CCC12CCOCC2 83582,N1(C(C(=O)Nc2scc(-c3ccc(CC)cc3)n2)=O)CCC12CCOC2 83583,C=C1CC(C(=O)NC23CC(c4ccccc4)(C2)C3)N(CCN2CCOCC2)C1 83584,CC(C)S(=O)(=O)C(C)C(=O)NCC(C)(C)NC(=O)Cn1cc([N+](=O)[O-])ccc1=O 83585,c1(OCC)oc(C)nc1C(=O)NC1CCCC1NC(C1(c2ccno2)CCC1)=O 83586,C#CC1CN(C(C2(NC(C3CC3(F)Cl)=O)CCSC2)=O)CCO1 83587,C1(C)(C(N(C)OC2CCCC2)=O)CCCN1C(C1COC(=O)N1)=O 83588,C1(CC(=O)NC2CCN(C(=O)CC3CC4(CC4)C3)C2)CC2(CCC2)C1 83589,c1(N2C(CCNC(Cc3cncc(C)c3)=O)CCC2)ccc2c(n1)CCC2=O 83590,C1(CNC(C(CCC)F)=O)N(C(=O)CN2CC(C)(OC)C2)CCCC1(C)C 83591,N1(C(CP(C)(C)=O)=O)CC2CCC2(NC(=O)Cc2ccc(Br)s2)C1 83592,C1(C(=O)NCc2ccc(C)s2)CCCN1S(=N)(=O)N(C)C 83593,N1(C(c2c(OC)n[nH]c2)=O)CCC(NC(C2CN(C)CCN(C)C2)=O)C12CCC2 83594,CC(C)C(F)C(=O)NC1(CNC(c2cscc2C#N)=O)CCOC1 83595,C(c1ccc(S(N)(=O)=O)cc1)=CC(=O)NC(CCNC(C(CC(C)C)C)=O)C 83596,CC1C(=O)NC(=O)CN1C(=O)C(CN=[N+]=[N-])NC(c1ccc(C(N)=O)o1)=O 83597,N1(C(C2N(C(C3C(C)CC=CC3)=O)C(C)C2)=O)CCCC12CCNC2=O 83598,c1(C(=O)NCC2CC(NC(CC(COC)(C)O)=O)C2)ccc(P(C)(C)=O)s1 83599,Cc1nnc(CNC(C2CCC(NC(C3CCCCC3)=O)C2)=O)o1 83600,C(=O)(C1=CCCOCC1)NC(C(C(=O)NC1(CC)CCOCC1)C)C 83601,C(=O)(C(CO)C(F)(F)F)NC1CN(C(c2cccc(C(C)(C)C)c2)=O)CC1SC 83602,CC1OCCC1(O)CNC(c1ccc(CNC(C23CSCC2C3)=O)nc1)=O 83603,c1(OC)ccc(CC(=O)NC2CCC2NC(c2sc(N)nc2C)=O)cc1F 83604,C1(C)(C(N2CC(CNC(c3n(CCC)nc(C)c3)=O)(OC)C2)=O)COCC1(F)F 83605,C=CCC(CNC(=O)C(C)(C)COC)C(=O)Nc1cncc(C(N)=O)c1 83606,CCCC(CCC)C(=O)NCC(c1ccccc1CC)NC(c1c[nH]nc1C)=O 83607,Cc1cnc(CC(=O)N(C(CNC(=O)CCCN2CCCCC2)C2CC2)C)s1 83608,N1(C(CCOCC(C)C)=O)CC(NC(C2C3CCCCCC23)=O)CC(F)C1 83609,CC(C)CCCCN(C(=O)C(n1cc(-c2cnc(C3CC3)s2)nn1)C)C 83610,C1(C(=O)NCC(CC)(CC)NC(=O)Cc2ccc(C)c(O)c2)CC12CCSCC2 83611,C(=O)(C(C)(F)C(F)(F)F)NCC(CC)NC(c1ncoc1-c1cc(C)no1)=O 83612,N12CC3(CC(F)(C1)C3)OC1CCN(CC1O)C2=O.C(C(F)(F)F)OC(C)(C)C 83613,Nc1c(C(=O)NC2C3CN(C(C4CC5CC5C4)=O)CC23)ccc(F)c1Cl 83614,C1(C(N2C(CNC(C3CC(OCC)C3)=O)CCCC2)=O)CCc2ncncc2C1 83615,c1(C(=O)NC2C(NC(=O)Cc3cncn3C3CC3)C2)cc2ccccn2n1 83616,N1(C(C=Cc2ccc(C)o2)=O)CC(NC(C2CN(c3nnnn3C)C2)=O)CC(C)C1 83617,Cc1ccccc1OCC(=O)NC1CC(C(=O)NCC(C)CO)C1 83618,C1(C)(CNC(COC(CC)C)=O)CCCN(C(c2cc(C(C)(C)C)n[nH]2)=O)C1 83619,N1(C(CN(CCCCC)C)=O)CCCC(C2(NC(=O)CCc3cn[nH]c3)CC2)C1 83620,O=C(CCCCC1CC1)NC1CN(C(C2(c3ccc(F)cc3)CCCCC2)=O)C1 83621,N1(C(CC2C(C)(C)C(O)C2)=O)CCCC(N=c2cc[nH]cc2[N+](=O)[O-])CC1 83622,C(=O)(C(=O)N=S(C)(C)=O)N1CCC(C)(NC(C2C(=C)CC2)=O)C1 83623,C1(C(N2C(C(=O)OC)C=CC2)=O)CN(C(c2cc(OC)no2)=O)CC1C 83624,C(=O)(C#CC1CCCCO1)NC1CC(CNC(C(C)NC(C)=O)=O)C1 83625,CC#CCCCC(=O)N1CCCC(CCNC(=O)CS(=O)(=O)NCC)CC1 83626,N1(C(c2c(C)oc(CO)c2)=O)CC2(CNC(=O)CN(C)CCO)CC(F)(C1)C2 83627,CCC(C)C(C(=O)NC1CCN(C(=O)C(F)C(C)(C)O)C(C)C1)OC 83628,c1(C(=O)OCC)nnc(N2CC(O)(C(C)NC(=O)CC3CSCCS3)C2)s1 83629,c1(C(C)NC(C2CCN(C(=O)CCCC3CC3C)C2)=O)nn(C)cc1O 83630,C1(NC(C(c2ccc(Cl)s2)C)=O)CN(C(c2cncc(O)c2)=O)CCC1CO 83631,C1(NC(CC(C)(C)C)=O)(CO)CCCN(C(=O)C(F)CC2CCCCC2)C1 83632,c1(OCC)cc(C(=O)NC2CC(NC(=O)CCCOC)C2)ccc1C 83633,C1(CC(=O)NCC2CN(C(=O)Nc3ccc(Cl)cc3)C3CC23)CN2CCC1CC2 83634,C12(NC(CN(C)C(=O)OC(C)(C)C)=O)CCC(NC(C3(Br)CCC3)=O)(CC1)CC2 83635,N1(C(C(N2CCC(C)C2)=O)=O)CCCC(C)(NC(c2cncc(N)c2)=O)C1 83636,c1(C(=O)NC2CC(N(C(=O)Cc3ccon3)C)C2)cnnn1C 83637,c1(CC(=O)NC2(C(N3CCC3C3CCCCC3)=O)CCOCC2)ccc(F)nc1 83638,CCCCCC(C)CC(=O)NC(CCN(C(=O)CCS(C)(=O)=O)C)C(C)C 83639,C1(CNC(CCC(N)=O)=O)(NC(C2CC(=O)N(CCO)C2)=O)CC2CCC1CC2 83640,c1(-c2cc(C(CC)C)no2)nc(-c2ccnc(Cl)c2)nn1C1CCCCC1 83641,CC1CN(C(C2C3CCC2(c2ccco2)C3)=O)CC1CNC(=O)CN(C)C 83642,C1(C2CN(C(=O)COc3cccc(Cl)c3Cl)C2)(NC(c2nc(C)nn2C)=O)CC1 83643,C1(CC=C)(C(=O)NC(C(C)C)c2ncc[nH]2)CCCN1C(c1ccncn1)=O 83644,c1(OC)cc(CNC(c2oc(CNC(c3cc(C)sn3)=O)nc2C)=O)ncn1 83645,CC1CC(C(=O)NC(C)(C)CN(C(=O)COc2ccc(CO)cc2)C)C(=O)O1 83646,C#CC(CNC(=O)CCCC(C)NC(c1nccnc1C)=O)CC(C)(C)C 83647,c1(C(C(=O)N2CCC2CNC(C2CCCSC2)=O)OCCC)ccc(F)cc1C 83648,C(=O)(C#CC1CCC1)N1CCC(CNC(CSc2n(C(C)(C)C)cnn2)=O)C1 83649,C(=O)(C1=NNC(C(F)(F)F)C1)N(CC(C)NC(CCC(=O)c1ccc(C)s1)=O)C 83650,N1(C(CCC(C)OC)=O)C2CCC1CC(N(C(=O)CCc1cc(C)no1)C)C2 83651,Cc1noc(N)c1C(=O)NCc1cc(C(=O)NC(C)Cc2ccccn2)n(C)n1 83652,C1(NC(c2cn(CC(N)=O)nn2)=O)CCSC12CN(C(C1CC3CCC1O3)=O)C2 83653,c1(C(N2CCC(C)(CNC(c3ccccc3)=O)C2)=O)cc(=O)c2ccccc2o1 83654,C1(OC)CN(C(c2ccc(C(C)C)cc2)=O)CC1NC(c1scnc1C)=O 83655,c1(OCC)ccc(C)nc1C(=O)NC(C)CN(C)C(c1[nH]ccc1CN(C)C)=O 83656,N#CC1CN(C(C2CCCN2Cc2cccc(O)c2OC(F)(F)F)=O)CCO1 83657,C(=O)(C1=CC2CCCCCCC12)NCCC(C)NC(=O)C(c1cccc(F)c1)C 83658,N1(C(C#CC(C)(C)O)=O)C2CCC1C(F)C(NC(c1cc(Cl)c([N+](=O)[O-])[nH]1)=O)C2 83659,C(C(=O)C(N)C(C)(C)C)NC(c1ccc(N(C)C)cc1)C 83660,N1(C(C(CSC)OC)=O)CCC(C=CC(=O)N(C)CCn2cccn2)CC1 83661,c1(C(N2C3CN(Cc4c(F)cccc4Br)CC23)=O)cc(F)c(F)c(O)c1F 83662,c1(CNC(c2n(C)cnc2Br)c2nnnn2CC(F)F)cccn2ccnc12 83663,c1(C(=O)NC(CNC(C2(CC)CCNC2=O)=O)CC(C)C)cccc(C)c1Cl 83664,Cc1occc1C1CC1C(=O)NCC1C=CCN1C(c1c[nH]c(=N)s1)=O 83665,Cc1nc(C)c(C(N2CC3(COC(CNC(C4CN(C)C4)=O)C3)C2)=O)c(C)n1 83666,CC1CN(C(=O)CS(=O)CC)CC1(C)C(=O)NCC(N1CCOCC1)=O 83667,C=CC1OCCC1NC(N1CCCC(C(=O)NCc2ccccc2)C1)=O 83668,N1(C(C=CS(C)=O)=O)C2CCC1CN(C(c1ncn3c1CCC3)=O)C2 83669,C1(C(=O)NCC2CC(C(C)C)C2)(NC(=O)C(C)c2cc[nH]n2)CCN(C)C1 83670,C(=O)(C1CCOc2ccccc21)O.N#CCC(C=O)OC(F)(F)F 83671,c1(C(=O)NC2(C)CN(C(C3CCCN(C)C3)=O)C2)cnn2ccn(C)c12 83672,c1(OC)cc(C)cc(C(=O)NC2(CN(C)C(C34CC3CNC4=O)=O)CC2)c1N 83673,N1(C(CC2(OC)CCC2)=O)CC(C)CN(C(c2cncc(C)c2Cl)=O)CC1C 83674,C(=O)(C(F)(F)CC(C)C)N(CC(CN(C(C(CC#C)C1CC1)=O)C)O)C 83675,N1(C(CO[Si](C)(C)C)=O)CC2(CCCC2CC(=O)Nc2cc3cc[nH]c3cn2)C1 83676,C1(C2CCC2)(CNC(C(C)(C)OCC)=O)CCN(C(c2cc(CO)on2)=O)CC1 83677,c1(C(N2CC(NC(c3n(C)cc(Cl)c3)=O)C(F)C2)=O)ccc2sncc2c1 83678,C(CC(CC)C(=O)N1CC(O)(C(C)(C)CNC(=O)COC(F)F)C1)=CC 83679,C1(C(N2C(C(C)(C)CNC(c3ccc(Cl)nc3)=O)CCC2)=O)CC2(C1)CC(O)C2 83680,N1(C(CCC(CC)NC(=O)Cc2cccs2)=O)CCN2C(=O)NCC2C1 83681,C(c1ccc(O)cc1)=CC(=O)NC(CNC(c1csc(-c2cn[nH]c2)n1)=O)CO 83682,Cc1cc(C)c(C#N)c(NC(C)CN(C)C(c2c[nH]cc(C)c2=O)=O)n1 83683,S(=O)(=O)(c1cccc(=NCC2CCOC(C)(C)C2)[nH]1)NCC1CCCN(C)C1=O 83684,C1(CNC(C(C)C2(O)CCC2)=O)CC(C(=O)N2CCOCC2C(N)=O)=NO1 83685,N1(C(C2N(CCC)CCCC2)=O)CCOC2(CCN(C(C34CCC3C4)=O)CC2)C1 83686,N1(C(C(COC)C)=O)CC(NC(c2cn3ncccc3n2)=O)CCC(O)C1 83687,c1(OC)nc(C(=O)NCCCC(C)(C)NC(=O)CN2CCC2C)sc1C 83688,C(C1CCCO1)=CC(=O)NC(C1CCN(C(=O)Cc2ccccn2)C1)C 83689,C1(C(C)(C2CC2)OC)CCN(N2CCn3c(C(C)C)cnc3C2)CC1 83690,Cc1cc([N+](=O)[O-])nn1C(C)C(=O)NC1CCN(C(=O)C=CCF)C1C(C)(C)C 83691,c1(N2C3CCN32)ccc(C(C2CCCOC2)=O)cc1.C(=O)(COC(C)(C)C)OC 83692,N#Cc1cccnc1NC1CC(NC(C2CCC(Cn3ccnn3)CC2)=O)C1 83693,c1(C(=O)NC2CCC(C)(CNC(CC=C=C)=O)C2)ccc2cc(F)ccc2n1 83694,c1(OC)cccc(NC(C2CCN(c3ccc(-c4cnoc4)nn3)CC2)=O)c1 83695,C(=O)(C1CCCc2nncn21)N(CCC)CCNC(=O)Cc1ccnc(O)c1 83696,c1(OC)cc(Cl)c(C)cc1C(N1CCC(NC(=O)CCc2ccccc2O)C1)=O 83697,c1(CCC)cc(C(=O)NC2CC3(C2)CC3NC(=O)C(O)C2CC2)nn1C 83698,N1(C(C(C)(C)C)=O)CC2CCCC2(Nc2cc3nncn3cn2)C1 83699,C1(NC(c2scc(COC)c2)=O)CC2CCC1(Cn1cc(-c3cc[nH]n3)nn1)C2 83700,C12(NC(c3c(C#N)ccs3)=O)CC3CCC(C1C2)N3C(=O)Cc1ccon1 83701,N12CCCC(C1)CCNC(=O)C2C.C(C)(C1CC1)=CC(=O)N(CC(=C)C)CCC 83702,C1(CCC(=O)NC(CC#C)CO)CCCCN1C(=O)Cc1csnn1 83703,CC1(C)OC(=O)CC1C(N1CC(NC(=O)CN2CCP(C)(=O)CC2)C2(CC2)C1)=O 83704,c1(COC)c(C(=O)N(C)C(c2cn(CC(O)CC)nn2)C)oc2ccccc12 83705,CCC(C)(C(=O)NC1CCCCC1NC(c1cnc(C(C)(C)C)s1)=O)OC 83706,c1(C(=O)NCC2C(NC(c3cc(Br)c[nH]3)=O)CCC2)cccn2c(O)nnc12 83707,CC(C(=O)NCCN(C(=O)CCC(F)(F)F)C1CCCCCC1)C(C)(C)C 83708,C1(COC)(CNC(=O)C(F)(F)CN(C)C)CCCN1C(C1CC(O)(C(F)F)C1)=O 83709,C(C(=O)NNC(=O)C(N)CC(F)F)N1CC(=O)N(Cc2cnn(C)n2)C1=O 83710,CC(Cl)(Cl)C(=O)NCC(CO)NC(C1CC1C(N)=O)=O 83711,c1(OC)nc(C(=O)NC2CC3CC2N(C(=O)C(N)=O)C3)cc2ccc(Br)cc12 83712,N(C1CC(C)n2ncnc21)C(C(=O)Nc1ccc(OC)c(-n2nnnc2C)c1)=O 83713,Cn1ncc(C(=O)NC2CCCC2CNC(c2cc[nH]c2)=O)c1F 83714,c1(C(=O)NCC(C)(CO)NC(c2n[nH]c(C)c2Br)=O)nccc(Cl)c1F 83715,N1(C(c2cc(CNC(C3(OC)CCCC3)=O)sc2)=O)CC(C(N)=O)OC(C)C1 83716,c1(OC)cccc(CNC(C2(NC(=O)CCC(C)C)CC2(C)C)=O)c1 83717,N#CC1(CC(N2CCCC(O)(CNC(=O)CC3CCC4CC34)C2)=O)CCOCC1 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83877,CCC(C)C(C(N)=O)n1cc(C2CN(C(=O)C(O)CC(C)C)CCN2C)nn1 83878,C=CC(C)(CCOC)C(=O)N(C)CCN(C(=O)C(c1ccc(C)cc1)C1CC1)C 83879,C1(C(=O)NC(C(C)C)C(=O)Nc2cnn(CCO)c2)CC2CC(=O)C1O2 83880,c1(NCC(=C)CC)nc2ccccc2nc1NCC(c1nncn1C)C 83881,C1(CNC(Cc2cc(C)ncc2)=O)CCN(C(=O)CC(C)C(F)F)C12CC2 83882,N1(C(CCCOCCC)=O)CC(NC(C2CCCNC2=O)=O)CC(F)C1 83883,C1(NC(=O)C=Cc2cncc(F)c2)CN(c2ncc([N+](=O)[O-])cn2)CC2(CC2)C1 83884,c1(C2(C(=O)NCCN(C)C(C34CCCC(CO3)C4)=O)CCCC2)ccc(F)cc1F 83885,N1(C(CC(C#CC)c2ccc(O)cc2)=O)CCCC2(CCCN2C(=O)C=C(C)C)C1 83886,C1(O)(CNC(C2C=CCN(C(C3C(C)(C)C3)=O)C2)=O)CCCCCC1 83887,Cc1cc(Cl)ccc1OCC(N1CCCOC(CNC(=O)C(C)(C)C(C)O)C1)=O 83888,C#CC(C1CCc2ccccc21)NC(=O)Nc1ccnc(C(F)(F)F)n1 83889,c1(CN(C(CN(C(=O)C2=CCCC2)CC#C)=O)C)ccc(C)nc1 83890,C1(CNC(C(C(C)C)OC)=O)CN(C(c2ncncc2Br)=O)CCC1C 83891,N1(C(C2(COC)CC2)=O)CC(NC(=O)CC23COC(C(=O)OC)(C2)C3)C2(CC2)C1 83892,c1(N2CC3C(C)(C)C(C3)C2)nc2ccccc2nc1NCC1CCCS1 83893,C=Cc1ccc(C(N2CC3CCC3(NC(=O)CC3CCN(C)C3=O)C2)=O)cc1 83894,N1(C(C(C)(C)C2CCCO2)=O)C2CCC(C2)C1C(N1CCC(N2CCCC2)C1)=O 83895,C1(NC(C=C(COC)C)=O)CC(NC(c2cc(O)cc(=O)o2)=O)C12CCC2 83896,C(CC(F)F)(C(=O)NC1CCC(O)CC1)NC(=O)CC1(O)CCC1 83897,c1(COC)nn(C)c(Cl)c1C(N1CCN(C(=O)CC2CC(C)=NO2)C(CO)C1)=O 83898,C1(C(C)C)CN(C(C2(C)CC2)=O)CCN1C(=O)CC1(c2ccc(Cl)cc2)CC1 83899,C1(CC(=O)NC2CC(NC(=O)CC3CCNC3=O)C2)CCCC1(F)F 83900,C1(C)(C(N2CC(C(C)NC(c3coc(CO)c3)=O)C2)=O)CC2CCC1C2 83901,c1(C(N(C(CNc2nccc(CC(=O)OC)n2)C)C)=O)coc2ccc(C)cc12 83902,c1(C(=O)NCC(C2CC2)NC(CCOC)=O)cc(-c2ccc(Cl)s2)on1 83903,C(=O)(C(C)C(C)NC(c1ncoc1C1CC1)=O)N(CC=C)CCOC 83904,C1(CNC(C(CC2CC2)OC)=O)CN(C(c2cc(C(N)=O)c[nH]2)=O)CC1O 83905,Cc1cc(C(=O)NCC(CC2CC2)C(=O)NC2CC2C(C)(C)C)ccc1F 83906,C1(CNC(CNC(=O)OC)=O)CC2CCC1N(C(=O)C(C)Cc1cccnc1)C2 83907,n1(CC(N2CC(OC)(CNC(c3ocnc3C)=O)C2)=O)cc([N+](=O)[O-])nc1C 83908,C1(C(N2CC(C)(CNC(C(C)C)=O)OCC2)=O)CCc2ncccc2C1 83909,C12(NC(CCN3CCN(CC)CC3)=O)CCCC1CN(C(c1cc(C)[nH]n1)=O)C2 83910,CCC(O)C(C)(C)C(=O)NCC1(CNC(=O)C=CC(=O)N(C)C)CCCC1 83911,C(=O)(CC(C(F)(F)F)NC(=O)CCC1(C)CC1)N(C1CC2CC2C1)C 83912,n1(CC(=O)NCCOCCN(C(CCC=C(C)C)=O)C)ncn(C)c1=O 83913,CCC(CC(F)(F)F)C(=O)NCC1(CCNC(=O)COCc2nc[nH]n2)CC1 83914,c1(C(=O)NC2C(F)CCN(C(C3ON=C(C)C3)=O)C2)c(C)nn2c1CCCC2 83915,c1(C(N2CCC2c2ccccc2)=O)cc2cccc(-c3ccc(CO)o3)c2[nH]1 83916,N1(C(c2ccc(C#C)c(C)c2)=O)CCC2CCC(C1)N2C(=O)Cn1ccnc1C 83917,N=c1nc(Cl)cc(C(=O)NCC2CCN(C(=O)Cc3ccc(Cl)cc3)CC2)[nH]1 83918,c1(C(=O)NC2C(CNC(c3cccs3)=O)CCCC2)cc2ccccc2[nH]1 83919,N(C(=NCCOCc1ccccc1)NC1CC=CC1)Cc1n(C)ncc1 83920,c1(C(=O)NC(C(N2C(C)CC2CO)=O)CO)ccc(N)cn1 83921,C(=O)(C(O)Cn1cncn1)NC(C)CN(C1CCCCC1)C 83922,c1(C(OCOC)C)cc(F)c(CNCc2cc(C)c(C)s2)cc1Br 83923,c1(C(C)C)cccc(C(N2CCOCC2CNC(C2CC3CC3C2)=O)=O)n1 83924,C(=O)(C#CC1CCOC1)NC(CC#C)C(=O)N(C1(c2cc[nH]n2)CC1)C 83925,C1(NC(=O)NCC(=O)NC(CN(C(C2CC2F)=O)CC)C)CCCCC1 83926,CC1C(C(=O)N(C)CCC2CC2)CCN1C(=O)Cc1ccccn1 83927,Cc1cc(=NCC23CC(NC(c4ncc(Cl)cc4Cl)=O)(C2)C(C)O3)c(C#N)c[nH]1 83928,N1(C(c2c(OC)nc(Cl)cc2)=O)CCCc2nc(Br)ccc21 83929,C1(CNC(=O)CSc2ccccc2O)CC12CCN(C(=O)C(O)C(F)(F)F)CC2 83930,C(=O)(C1=CC=CN2CCS(=O)(=O)N=C12)NCC1(NC(CP(C)(C)=O)=O)CCOC1 83931,N1(C(c2nn(C)cc2Br)C(=O)NCC(=C)C)CC(S(C)(=O)=O)CCC1C 83932,c1(C(=O)NC2CCCC(NC(CCc3cc(C)sc3C)=O)C2)ccnc(C)c1N 83933,[N-]=[N+]=Nc1cccc(C(=O)NCC2CCCC2NC(=O)CCc2cc(Cl)cs2)c1 83934,c1(CN(C(c2cnn(CC(F)F)c2)C(=O)NC2CCC2)C)cc2ccccc2s1 83935,c1(SC)ccc(C(N2CCCC2CC(=O)NCC(=O)NCC(F)F)=O)o1 83936,CC(C)CC(C)CC(=O)N1CCN(CCOc2cc(O)ccc2OC(F)F)CC1 83937,C1(C(N2C(CCNC(C(CCCOC)C)=O)CCCC2)=O)CC1C1CCCCC1 83938,C(N=c1cc(Cl)nc(C2CC2)[nH]1)C1OCCN(C(C2CCC(C)(C)OC2)=O)C1 83939,N1(C(c2n(CCOC)ncc2)=O)CCC(CNC(c2ncc(Cl)n2C)=O)C(C)C1 83940,C1(CC)CN(C(c2c(Cl)noc2C)=O)CC1NC(=O)C(c1ccccc1)F 83941,C1(N(C)C(C2CCC3(CC3)C2)=O)CN(C(C2CC2c2cnn(C)c2)=O)CCC1O 83942,Cc1ccccc1C=CC(N1CCC(C)(CNC(C2C3COCC23)=O)C1)=O 83943,c1(-c2cn(CC=C)nc2)cnc2[nH]cc(C(=O)Nc3[nH]cnc3CC)c2c1 83944,c1(OC)cccc(-n2nnnc2C2(NCC3CC4CCC3O4)COC(C)C2)c1 83945,C(CCCN=c1[nH]c(Cl)nc2c1SCC2)NC(C(CCCC)O)=O 83946,Cn1nc(C(=O)NC2CC2NC(c2ncsc2C(F)(F)F)=O)ccc1=O 83947,Cc1cc(C)c(C(N2CC=CC(NC(=O)CCCc3csc(C)n3)C2)=O)c(N)c1 83948,Cn1c(C(N2CCC(CCC(N3CCC(F)(CF)C3)=O)C2)=O)nnc1S 83949,c1(CCC(=O)N(CC(C)NC(CCC=C(C)C)=O)C)cccc(C#N)c1 83950,n1(C(C)C)cncc1C(=O)OCC1CC=CCO1 83951,c1(NC(=O)NC2CC(NC(C3CC(C(F)F)C3)=O)C2)ccccc1Br 83952,N1(C(c2cc(C)[nH]n2)=O)CC2CC(C1)N(C(C1CCC(C)(C)O1)=O)C2 83953,CCCCCC(C(=O)NC1CC1NC(c1cc2sc(N(C)C)nc2s1)=O)C(C)C 83954,N1(C(C2CC(C)=C(C)CC2)=O)CC(CNC(=O)C=CC2CCCC2)CC12CCC2 83955,C#CCC(C)(C(=O)NC(C)CCC(=C)C)NC(=O)Cn1nnnc1C 83956,N1(C(C2(C(=O)OCC)CC2)=O)CC(CNC(=O)COC(F)F)C1 83957,c1(C(=O)NCC2C(NC(CC(=O)OC)=O)CC2)nc(OC)ccc1OC 83958,Cc1cc(NCCC2CCC(NC(C3(C)CCCOC3)=O)C2)ccc1[N+](=O)[O-] 83959,c1(C(N2CCC(SC(F)(F)F)CC2)C(=O)NCCCCCC)cc(C)nnc1C 83960,Cc1ccc(C2CC2C(=O)NCC2(NC(=O)CC(C)C(C)C)CCC2)c(Cl)n1 83961,Cc1c(C(=O)NC2CC2NC(=O)CC2CCCO2)cccc1C#N 83962,N1(C(c2c(F)ccc(C)c2)=O)CCCN(C(c2cc(Cl)cs2)=O)CC1C 83963,Cc1cnc2c(C(N3CC(NC(=O)Cn4cnc(=N)[nH]4)CC(F)C3)=O)cccn12 83964,C1(CNC(CC2(N(C(C(COC)(C)O)=O)C)CC2)=O)CC(C(N)=O)=NO1 83965,N1(C(=O)OC(C)(C)C)C2CCC(C2)C1CNc1ccc(CCF)cc1 83966,c1(C(=O)NC2CC(NC(c3cc(Cl)c(Cl)cn3)=O)C2)cnc2cc(Cl)ccn12 83967,C12(C(N3CCCC(CC=C)(NC(=O)C=CC(C)C)C3)=O)CCC(C#N)(CC1)CC2 83968,CC(CC(=O)NC1CS(=O)C1)N(C(=O)CCc1ccn(C)n1)C 83969,c1(SCC)ccc(Br)cc1C(N1CCCCC1C1CCN(C(C)=O)C1)=O 83970,C(CCCCCCC(=O)NC1CC2CN(C(c3occc3Cl)=O)CC2C1)SC 83971,O=C(N1CC(n2cc(-c3ccc(N)cn3)nn2)CO1)C1CC2(C1)CC2(F)F 83972,C(=O)(C(CCC)C(C)C)NCCC1CCCN(C(C(CCC)F)=O)CC1 83973,C(=O)(CC(C)(C)OC)N(CCCCCNC(C1CCN(C(CC)CC)C1)=O)CC 83974,C1(C(=O)NOCC(C)C)(CCOCC)CCN(C(c2cnn(C)c2)=O)CC1 83975,C(=O)(C(C)(C)C(C)(F)F)NC(=O)C(CC(N)=O)N(C)C(C)=O.CC(CN)OC(C)(C)C 83976,C(=O)(CCCCC(F)F)NCC1CCC(N(C(c2cnn(C)c(=O)c2)=O)C)CC1 83977,c1(C(N(CCN(C(C2CC(CC(C)(C)C)C2)=O)CC)CC)=O)ccc(Br)nc1N 83978,C1(C(N2CC(OC)CC(NC(CCC#C)=O)C2)=O)CC(C(C)(C)C)=NO1 83979,c1(C(=O)NCC(CC=C)NC(=O)C(O)CN(C)C)ccc(Cl)cc1C 83980,c1(C2(C(N(CCC)CCOC)=O)CC2)ccc(OC(F)F)cc1 83981,N1(C(c2c(C)n(C)nn2)=O)CCN(C(c2ccnn2C)=O)CC1c1cccnc1 83982,CC(C(=O)NC1C2CC1CN(C(c1ccnn1C1CCOCC1)=O)C2)C(C)(C)C 83983,CC1(C)CCN(C(=O)C=C2CCCCC2)CC1NC(=O)CC1CCCOC1 83984,C=CCC(C)(C)CC(=O)N1C(C)C2CC1C2NC(c1cnc(O)n1C)=O 83985,C1(CC(C)NC(=O)C=CC(C)(C)C)CCN(C(C2CC2c2nncn2C)=O)CC1 83986,CN1CCN(CCC(=O)NC(C)(C)CN2CCN(C(C3CCOC3)=O)CC2)CC1 83987,c1(C(=O)NCC2C(C)CN(C(c3cccc(Cl)c3)=O)C2)cc2cnn(C)c2s1 83988,CC(CC(=O)NC1CCCC(NC(c2ccn(C)c(=O)c2)=O)C1)CC(F)(F)F 83989,N1(C(CC(C(C)C)O)=O)CCC2(CCCCN(C(c3cn(C)c(=O)cn3)=O)C2)C1 83990,C(C)(CNC(=O)C(C)C(C)(F)F)(CC(C)C)NC(CCNC(C(C)C)=O)=O 83991,c1(C(N2C(CCC(=O)NCCC(=C)C)CCCC2)=O)n[nH]cc1[N+](=O)[O-] 83992,c1(CN2CC(C(=O)Nc3ccc(CC)nc3)OCC2)ccc(I)c(O)c1 83993,C=CCC(CC(=O)NC(C)C(CC)CC)NC(=O)Cc1ccc(C)s1 83994,c1(C(N(CCOC)CCNC(=O)C(F)(F)CN(C)C)=O)sc(C)c(C)c1C 83995,C(=O)(C1CCCc2nncn21)N1CC(CNC(C(CCC(C)C)NC(C)=O)=O)C1 83996,C1(NC(C(F)=CC)=O)CN(C(c2ccc(-c3cccnc3)cn2)=O)CC1(C)C 83997,C1(C(=O)NCCCN(C(=O)CCC(=O)c2ccc[nH]2)C)CC1C1CCCCC1 83998,c1(C(=O)NC2C3CN(C(c4c(C)ncnc4)=O)CC32)ccc2nn[nH]c2c1 83999,CC1(C)CCCCC1=CC(N1CC(CNC(C2C3CCCOC23)=O)C(O)C1)=O 84000,N1(CCC)CC(C(N2CC(CN(c3ncc(C(F)F)cn3)C)C2)=O)CC1=O 84001,C1(O)(C(=O)NC2CC(CCNC(c3cc(OC)n[nH]3)=O)C2)CC2(CCOCC2)C1 84002,C1(C(=O)NC(C2CCOCC2)C#C)CCN(C(c2ccsn2)=O)CC1O 84003,Cc1noc2cc(C(N3CC(CCNC(=O)CN(C)CCO)C(C)C3)=O)ccc12 84004,CCCC(CC(C)C)C(=O)N1CCOCC(NC(c2occc2COCC)=O)C1 84005,c1(C(=O)NCc2cccc(CNC(CCCSC)=O)c2)c(C)cc(C)cc1N 84006,CC1CCN(C(C2CC(=O)N(C)C2)=O)CCN1C(=O)CCN1CCCCC1=O 84007,N1(C(C2N(CC)C(=O)CC2)=O)CCCC2(CCN(C(=O)CN3CCC(C)C3)C2)C1 84008,C(CC(C(C)C)NC(c1nccnc1C(N)=O)=O)NC(C(C)=C(C)C)=O 84009,CC(C)CC(CNC(=O)CC1(C)CC1)NC(c1ccc(C2CC2)o1)=O 84010,c1(OCC)ccc(-c2nc(COC)nn2-c2ccnn2C)cc1OC 84011,C(C)(CO)(C(=O)N1CCOC(C2CN(C(=O)Cn3cc(C)cn3)C2)C1)NC(=O)OC 84012,CC(C)(C)[Si](C)(C)OCC1(F)CN(C(c2cnc(C#N)nc2)=O)C1 84013,N1(CC(N2CCC(O)(CN(C)C(c3cn(C)nn3)=O)C2)=O)CCCCCC1=O 84014,c1(NC2CCN(C(CC)C)CC2)[nH]c(=NCC(CC)C(C)(F)F)nc2sccc12 84015,c1(NC(N2CC(C(C(=O)OCC)C)C2)=O)cc(COC)no1 84016,C(=O)(C(C)C(C)(C)C)N(C(CNC(C(c1ccccc1O)OC)=O)C)C 84017,N1(C(C(C)OC)=O)CC2CCC(C1)C2C(N1CCCC1c1ccccc1)=O 84018,c1(C(N(CC(CNC(C(c2cccc(C)c2)=O)=O)O)C)=O)cc2sccc2n1C 84019,Cc1cc(C(=O)NCC2C3CCC(C3)N2C(=O)CCc2cnn(C)c2)c(C)cn1 84020,C(=O)(C(C)(C)CC(F)F)NC1CCN(C(c2cnn(C)c2C(F)F)=O)C1C1CC1 84021,C(C(N=c1nc(C2CC2)[nH]s1)C1CC1)N(CC(F)F)C(c1onc2c1CCCC2)=O 84022,C#CCCN=C(NCCOC1CCS(=O)(=O)C1)NCc1cnn(C)n1 84023,C1(CNC(Cn2ccc(C)n2)=O)CC2CN(C(=O)C(c3ccc(F)cc3)F)CC12 84024,N1(C(COCC=C)=O)Cc2n[nH]cc2C1C(=O)N(C1CCCCCC1)C 84025,C(c1c(OC)cnn1CC=C)=CC(=O)NCC1N(C(CC(C=C)C)=O)CC(O)C1 84026,c1(C(=O)NCc2c(C(=O)NCC(CCC)O)n[nH]c2)c[nH]ccc1=O 84027,c1(CCC(N2CCC(n3cc(C(COC)OC)nn3)C2)=O)cccc(N(C)C)c1 84028,c1(CN2CCC(O)(Cc3ccccc3)C2)noc2c1COCC2 84029,CCC(C)CCCC(=O)NC(C1CCCN1C(=O)CSCc1ncc[nH]1)(C)C 84030,N1(C(C2C(=C)C2C(=O)OC)=O)CCN(C(C23CCOC(C)(C2)C3)=O)C(C)C1 84031,c1(C(=O)NCC(CN(C(c2cc(C)no2)=O)C)O)ccc(N)c(C)c1C 84032,O=C(C1=CCCOCC1)NCC1CC2CC2N1C(=O)C=Cc1ccc(F)c(Cl)c1 84033,c1(NC(CC2(C=C)CN(C(=O)C(C)CSC)C2)=O)ccc(F)c(CC)c1 84034,N1(C(c2n[nH]c(C)c2[N+](=O)[O-])=O)CCc2ccc(N=[N+]=[N-])cc2C1 84035,N1(C(c2c(CC)nn[nH]2)=O)CCC(CF)(NC(=O)CCCN(C)C)C1 84036,CC1CN(C(C2(C#N)CCCC2)=O)CCC1N(C(=O)C1=NOCC1)C 84037,N1(C(CC(C)(C)O)=O)CCN(C(C2CC2c2ccc(Cl)c(F)c2)=O)CC1CCO 84038,c1(C(=O)NC(CC=C)CNC(=O)Cc2nc[nH]n2)ccc(C=NOC)cc1 84039,C(C)(c1ccc(F)cc1)=CC(=O)NC(C1(O)CCN(C(C(C(CC)O)C)=O)C1)C 84040,c1(C(=O)NCC2C(NC(C(c3ccccc3F)OC)=O)C2)cc(C#N)[nH]c1C 84041,N1(C(CCOCCC)=O)CC(NC(=O)Cc2cc(F)c(N)cc2F)CC2(CC2)C1 84042,C1(CCNC(C(CC)O)=O)CN(C(c2cc(Br)cn2C(C)C)=O)CCO1 84043,CC(O)C(C(=O)N1CCC(CCNC(=O)C(c2ccccc2F)O)CC1)N(C)C 84044,C1(C)(CC)C=C(C(=O)N2CC(CNC(c3cc(C(C)=O)oc3C)=O)C(F)(F)C2)C1 84045,N1(C(c2nc(C)oc2C)=O)CC(C)(C)CC1CNC(=O)C=CC1CCCN1C 84046,CC(CC(=O)NCCC(O)CCO)C(C)(C)NC(=O)C(CO)C(C)(C)C 84047,c1(OC)cc(C(N2CC(NC(c3cc(C)no3)=O)CC2(C)C)=O)c(F)cn1 84048,C(CNC(=O)C(c1ccccc1Br)O)(C(C)(C)C)NC(C(C)N(C)C)=O 84049,N1(c2n(CCOCC)nnn2)CCOCC(CCC2CC2)C1.c12ccc(cc1)s2 84050,N1(C(C(CC)CCOC)=O)CCC(C2CC2)(NC(c2cncc(F)c2Cl)=O)C1 84051,C1(NC(Cc2cc(C)c(CO)cc2)=O)CCCC12CCN(C(=O)C(N)=O)C2 84052,Cc1nn2ccccc2c1C(=O)NCC1(CCNC(C2(C)CC=CCC2)=O)CC1 84053,N1(C(C(C)OCC)=O)CCC2(CCC2NC(=O)CC=Cc2ccccc2)CC1 84054,N1(C(C=C(CC)C)=O)CCC2(CC1)CCN(C(=O)C(C)(C)CF)CC2C 84055,c1(C(C)C)c(C(=O)NC2CCCCC2NC(=O)C(C)n2cccn2)cccc1F 84056,CC1CC(NC(=O)Cn2ccc(O)nc2=O)CN(C(=O)CNS(=O)(=O)N(C)C)C1 84057,C1(NC(c2c(C)coc2)=O)C2CCCN(C(C3OC4CCC3C4)=O)C2C1(C)C 84058,C1(C(N(C)Cc2c(OC)ccc(CO)c2)=O)C2CCCC(F)(F)C12 84059,n1(CCCC(=O)NCC(CNC(CC2(C)CC2(Cl)Cl)=O)CO)ccccc1=O 84060,c1(C(N2CCCC(NC(c3c(C)ncn3O)=O)C2)=O)cc([N+](=O)[O-])c[nH]1 84061,C1(C(=O)Nc2ccc(C(C)(C)C#N)cc2)CC2C(C1)C2(F)F 84062,c1(CNC(C(CC)F)=O)cccc(NC(=O)CC(C)CNS(=O)(=O)C(C)C)c1 84063,c1(-c2ccc(OCCC)cc2C)ccc2cc(C(=O)Nc3cnnn3C)[nH]c2n1 84064,N1(C(C2=CC(C)CC2)=O)CCC2(CCN(C(c3ccc4cc[nH]c4n3)=O)C2)C1 84065,c1(C(=O)NC(CC)CN(C(C2CCC(CCO)CC2)=O)CC)cnc(O)c(F)c1 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84169,C=CCCC(C(=O)NCC1CC(OC)C1)NC(C1CC12CCOCC2)=O 84170,CCCCC(CC)NC(C1CSCCN1C(c1cc(CO)c(C)o1)=O)=O 84171,N1(C(C(C)(C)NC(C2(CC(=O)OC)CC2)=O)=O)CC(S(C)(=N)=O)C1 84172,N1(C(C(C)NC(=O)NC(C)(C)C)=O)CCC(CO)C(C)(C)C1 84173,C1(CCN)(OC)CCCN(C(C2(C3(c4ccccc4)NC(=O)NC3=O)CC2)=O)C1 84174,c1(C(=O)NCC2C(NC(=O)COCC(F)(F)F)C2)n[nH]c(C2CC2)c1Br 84175,c1(C(=O)NC2C(NC(CSCCC(C)C)=O)CC2)n[nH]cc1-c1ccncc1 84176,N1(C(=O)C2CC2)CCN2CCN(C(=O)COC3CCCC(=O)N3)CC2C1 84177,N1(C(c2ccc(P(C)(C)=O)o2)=O)CCC2CN(C(=O)COC(F)F)CCC2C1 84178,N1(C(C2C(NC(C3C(C(=O)OC)C=C3)=O)CCO2)=O)CCN(C)CC1C 84179,N(C(=NCCCC(=O)N1CCCC1)NCC12CCCC1CCO2)CC(C)C 84180,c1(C(=O)NC(CNC(c2ccc(=N)[nH]c2)=O)C2CC2)ccc2cnnn2c1 84181,C(=O)(CC(C)NC(=O)CC1CC=CCC1)NCCOCCOCC 84182,Cc1nn(Cc2nc(-c3cccc(COC(C)(C)C)n3)nn2C)c2ncccc12 84183,N1(c2nc(C3(NC(=O)CCc4cn(CCCF)nn4)CC3)on2)CCCCCC1 84184,c1(CC(C(=O)NC2CC(N(C(=O)CCF)C)C2)OC)ccc(C)cc1 84185,Cc1cc(C(=O)NC2(CC(=O)NCC(C)(C)CCO)CCCCC2)ccc1O 84186,C1(CC)(CC)CN(C(C23CCC(C2)C3OC)=O)CC(C)O1 84187,C(C(=O)N1CC(NC(c2cc(O)n(C)n2)=O)CC1(C)C)(C(C)(C)C)NC(C)=O 84188,C(C)(C)(CCCC(=O)N1CCOCC1)NC(CC1CCN(C)CC1)=O 84189,N1(C(CC2C(C)CCC2)=O)CCC(CCNC(C2(n3cc(Cl)cn3)CC2)=O)CC1 84190,CCC(CC)CCC(=O)NCCCN(CCCCNC(c1cccn1C)=O)C 84191,Cc1ccc(C(=O)NC2CCC(NCc3cc(C(=O)O)ccc3F)C2)cc1Cl 84192,N1(c2n[nH]c(=Nc3cnn(C)c3Cl)s2)CCC2(CC1)CCS(=O)(=O)CC2 84193,N1(C(c2c(C)c[nH]c2)=O)CCc2cc(C(=O)NCC(N)=O)cnc2C1 84194,C1(CC)(CO)CC(NC(=O)C(=O)NC2(c3nc(C)cs3)CCCC2)C1 84195,N1(C(C#CC2(C)COC2)=O)CCC2CCN(C(=O)CCc3ncc(F)cn3)C2C1 84196,N1(C(C)C)CCCC(CCNC(C2CCCCN2C(=O)COC2CC=CC2)=O)C1 84197,C=CCC(CC(C)C)C(=O)NCC(CCC)C(=O)NCc1ncc(F)cc1F 84198,CC(CC(=O)N1CC2OCC(NC(C3COCCOC3)=O)C2C1)CC(C)(C)C 84199,C=CC(C)(C)CC(=O)N(CCN(C(C1CC(O)CN1C)=O)CC)CC 84200,C(=O)(CCCN(C)N=O)NCCC1OCCN(C(CC2C(C)CCCC2)=O)C1 84201,c1(C(N2C3CN(C(c4c(OC)cccn4)=O)C(C3)C2)=O)oc2ccccc2c1C 84202,C1(C(N(C2(C(=O)NCc3nccc(C)c3)CC2)C)=O)C2CCC(C2)C1C 84203,C(C)(CNC(C1(c2ccnn2C)CC1)=O)(C(C)C)NC(c1c(SC)ccs1)=O 84204,N1(C(C2(C#C)CCCCC2)=O)CCC2CC2(C(=O)NC(CO)C(O)CCC)CC1 84205,CC1=CCC=CC1C(N1CC2C(NC(=O)CC(C)O)C2C1)=O 84206,S(=O)(=O)(C1(Cc2cccc(Cl)c2)CC1)N(C)C.N12CCC(C1)CCNC2 84207,N1(C(C(C)n2cccn2)=O)CCC(CNC(C2C3CCC23)=O)CC1 84208,C1(NC(CN2CCC(C(N)=O)CC2)=O)CC2CCC(C1)N2C(c1ccnnc1)=O 84209,N1(c2nc(OC)c(F)c(C)n2)CCCC2(CCN(C(=O)C(C)(C)SC)C2)C1 84210,C1(C(NOCCCCCC)=O)CCCN(C(=O)Cc2cnccc2C)C1 84211,N1(C(C(CC)OCC)=O)CCN(C(c2cnc(O)nc2O)=O)CCC1C 84212,C(=O)(C(C)(C)C(N)=O)N(CCC(C)NC(c1cnn(C(C)C)n1)=O)C 84213,N1(C(C(C(C)C)NC(=O)OC)=O)CCC(F)(CNC(=O)C(F)CC(C)C)CC1 84214,n1(C(C)C)cnc(C(=O)NC2CCC(NC(=O)C(=O)NC(C)C)C2)c1 84215,C=CCC(CC(C)C)C(=O)N1CCOC2(C1)CN(C(=O)COCCN(C)C)C2 84216,c1(NC(C)=O)ccc(C(N2CCCC(N(C)C(c3cccn3C)=O)C2)=O)cc1F 84217,C1(NC(=O)OCC)CCN(N2CCC(OCc3ccc(F)cc3)C2)CC1 84218,CN1CC(C(=O)NCCCN(C(C2CCCS2)=O)CC2CCCC2)CC1=O 84219,c1(C(N(CCNC(C2CC3CCC3C2)=O)CC2CC2)=O)cc(F)cc2nc[nH]c12 84220,c1(C(N2C(CNC(CCC=CCC=C)=O)COCC2)=O)cc(F)cc(C)c1N 84221,Cc1cc(C(C)NC(C2CCN(C(c3ccnnc3)=O)C2)=O)on1 84222,CCCC(CC1CCCC1)C(=O)N1CCCC(NC(=O)CC2(C)CCOCC2)C1C 84223,C(=O)(CCC(C)(C)[N+](=O)[O-])N(C(C)C(=O)NCCc1ccns1)C1CC1 84224,C(=O)(CCCCC(=O)NCC(O)CN(C(=O)C(O)C1=CCCCC1)C)OC 84225,CN1CCC(=CC(N2CC3C(CNC(=O)CCC4(C)CC4)C3C2)=O)CC1 84226,Cc1csc2c(NCC3CN(C(=O)C(C)(C)CO)CC34CCC4)ncnc12 84227,c1(CC)ccc(C(C(=O)NC)NC(=O)CN(CCOC)CCOC)nc1.C1(C)CC1 84228,C(CC(O)C(=O)OC)NC(CCN(C(C=CC)=O)CC)=O 84229,c1(CCC(=O)NC(C2(O)CN(C(C3(CC=C)CC3)=O)C2)C)ccc(Cl)cc1 84230,C(=O)(CC(C)C(C)(C)NC(=O)C1=CCCOC1)Nc1ccc(CC)cc1C 84231,C(CN=C(NCCF)N1CCC(O)(c2ccc(F)cc2)C1)=CCC 84232,N1(C(c2cc(-c3ccco3)[nH]n2)=O)CC2CCC(C1)N2C(C1(CC(F)(F)F)CC1)=O 84233,c1(C(N2CCCC2c2cccc(Cl)c2)=O)cc(Cl)c(F)cc1[N+](=O)[O-] 84234,c1(CC(=O)NC2CCN(C(c3c(C)ncnc3)=O)C2)cnn2c1OCCC2 84235,N1(C(C2CCCC(C(C)C)C2)=O)CC2=C(C1)CN(C(c1cc(F)cc(Cl)c1)=O)C2 84236,c1(OC(C(=O)NCCN(C(=O)C(O)C(C)C)CCC)C)cccc(C(C)=O)c1 84237,CC(C(F)(F)C(F)(F)F)NC(=O)C(C1CCCN(C(=O)OC(C)(C)C)C1)(F)F 84238,C(=O)(C(Cc1ccco1)NC(=O)CCC1CCCOC1)N(CC=C)C 84239,N1(C(CN(C(CCOC)=O)C)=O)CCN(C(=O)CCCCCSC)CC1CCO 84240,c1(CC)cc(C(=O)N(C2CCN(C(=O)CCc3cncc(F)c3)CC2)C)c(C)o1 84241,c1(CN2CC(n3ncc(NC(c4ccnc(O)c4)=O)c3)C2)cccc2c1CCC2 84242,C(CC(CNC(C1(C)CC(F)C1)=O)NC(=O)COCCF)OC 84243,c1(CC(N2CC3CC(CNC(C4(C)CC4)=O)C3C2)=O)ccc2ncsc2c1 84244,N1(C(C2N(CC)CCOC2)=O)CCC2OCCN(C(=O)CC(C)(C)OC)C2C1 84245,C1(CC(=O)N(C2CCN(C(=O)C(C)CC3CC3)C2)CC#C)CSCCO1 84246,C12(CNC(C(C)c3ccsc3)=O)CCCC(CN1C(=O)C=Cc1cncs1)C2 84247,C1(C(=O)NC2CN(C(c3cc(SC)oc3C)=O)CC2C)(OC)CCOCC1 84248,S(=O)(=O)(C1CC1)NC(c1ccccc1)C(=O)NC1CC(O)C1 84249,c1(CCC(=O)NC2CN(C(C3(c4ccnnc4)CC3)=O)C2)ccc(OCF)cc1 84250,c1(C(=O)NCC(CNC(C(C)OCC=C)=O)CO)cc(F)ccc1NS(C)(=O)=O 84251,C1(CNC(N(C2CCCN(C)C2)C)=O)CCCN2CCCCC12 84252,CC(C)CCCCC(=O)NC1(C)CC(NC(c2cnn(-c3ccccn3)c2)=O)C1 84253,c1(CC)c(C(=O)N(C(C)C(=O)NCCC(C(=O)OC)OC)CC)nnn1C 84254,C(=O)(CC(CC(C)C)NC(C1CCOC1)=O)N1CC(c2onc(C)n2)C1 84255,C1(N(C)CC)CCCCC1NC(=O)NC1CCCN(C(=O)NC)C1 84256,N1(C(CN2CCN(C(C(C)n3ccnn3)=O)CC2)=O)CC2CCCCC2C1C 84257,C(C)(CNC(c1c[nH]nc1C(F)F)=O)(C(C)C)NC(C(CO)OC)=O 84258,C1(N(C)C)CCC(C(=O)NC2C3CC2N(C(C2(C)CC=CC2)=O)C3)CC1 84259,c1(NCc2c(OC)ncc(F)c2)cnc2ccc(F)cc2c1 84260,N(C(=NCCF)N(C)Cc1cc(Cl)ccc1Br)C1CCC(C(C)C)C1 84261,C1(n2cc(COC)nn2)CCCCC1C(=O)NCc1ccccc1Cl 84262,c1(OC)c(C(=O)NC2CC2CNC(C2(C)CCC3CC3C2)=O)c(C)nn1C 84263,C1(O)(C(C)C)CCCN(C(C2CC3C=CC2CC3)=O)C1 84264,CCC(COC)(CC)C(=O)N1CCC(C(=O)N(C2CCOC2)C)O1 84265,N1(C(c2c[nH]c(=NC)s2)=O)CCC2(CC1)CC2C(N1CCOC(C(C)(C)C)C1)=O 84266,c1(C(N2C(C)CC(NC(C3(Br)CC3)=O)C2)=O)cc(-n2ccnc2)ccc1O 84267,Cc1c(CC(N2CCC(C(C)NC(c3ccc(C(F)F)o3)=O)CC2)=O)nnn1C 84268,C1(COC)(NC(C2(n3cccn3)CC2)=O)CCN(C(=O)CCn2cncn2)C1 84269,C1(C(=O)NCC(CNC(c2cc(C)ns2)=O)CO)CCC(=O)NC1 84270,C(=O)(C(C)(C)C(N)=O)N1CCN(CC(C)NC(c2cnc(O)c(F)c2)=O)CC1 84271,N1(c2nnc(C(N)=O)s2)CC2C3CCC(C2C1)N(C(C1(CC2CC2)CC1)=O)C3 84272,CC(=O)CC(C)(C)C(=O)NCC1CC(C(=O)NCC(C)CC2CCC2)C1 84273,C1(C(N(CCCC=C)CC)=O)CCC(C2CC2)N1C(=O)C=Cc1cc[nH]n1 84274,c1(C(=O)NCC2CCCC2C(N2CC(n3cccn3)C2)=O)ccncc1F 84275,c1(C(N2CC(NC(C3(CC#C)CCC3)=O)C(F)C2)=O)cnc2n1CCOC2 84276,C(CO)(CCCCNC(=O)CC(C)c1cccnc1)NC(c1nc(CC)sc1)=O 84277,c1(C(N2CC=CC(NC(CC3COCC(C)O3)=O)C2)=O)cccc(F)c1F 84278,C(CCCCNC(=O)CCCF)NC(C(C)c1cccs1)=O 84279,C1(C(=O)NCC2(CCC)CC2)CCCCN(C(=O)C(C)(CO)OC)C1 84280,C(=O)(C1=CCOCC1)NC(C1(O)CCN(C(=O)CC2SC(=N)NC2=O)C1)C 84281,n12cc(nn1)C2.N1(CC2CN(C(C3CCC3)=O)C2)CCOC1=O 84282,c1(CNC(CNC(=O)NC)=O)ocnc1C(=O)NCCC1CCN(C)C1 84283,Cc1ccc(C(N2CCCOC(CNC(=O)C(C)NC=O)C2)=O)c2c1CCC2 84284,N1(C(C(N2CCC(c3ccc(N(C)C)cc3)CC2)C)=O)CCN(C)CC1 84285,c1(NC(C)=O)ccc(SCCC(=O)NC2CC(NC(=O)C=CSC)C2)cc1C 84286,C(=O)(C(C(C)(C)C)C1CCCCC1)N(C)CCNC(c1cn(C)[nH]c1=N)=O 84287,CC1CN(C(C2CC(c3ccccc3)C2)=O)CCN1C(c1ccc(O)nc1Cl)=O 84288,CCCC(C)C(=O)NC1CCCN(C(C2(C#N)CCC2)=O)C1 84289,Cc1cc(F)c(CN2CCCC2CNC(c2csc3c2CCCC3)=O)cc1Br 84290,CCC(CNC(=O)C(c1cncnc1)C)(CC)C(=O)NCC(O)C1(Cl)CC1 84291,Cc1scc(C(=O)NC(C2(O)CCN(C(=O)CC3CCOCC3)C2)C)c1C 84292,CC1(C)COC(CCC(=O)NCCN(C(=O)CCOCC(F)F)C2CC2)C1 84293,c1(NC(C2C3CN(S(c4ccn(C)n4)(=O)=O)CC32)=O)cc(F)cc2[nH]ncc12 84294,Cc1cc2[nH]c(C(=O)NCC3(CNC(=O)CNC(=O)C4CC4)CC34CCC4)cc2o1 84295,C(CC(C(=O)N(C)Cc1nnnn1C)NC(C1CC(OC)C1)=O)OC 84296,C12(NC(=O)Cc3ccc(F)cc3Cl)CCCC1N(Cc1cccc(Cl)c1Cl)CC2 84297,N#Cc1ccc(CC(=O)NCCOC2CCN(c3ncc(Br)cn3)C2)cc1 84298,CC(O)C(C)(C)CNC(=O)C(F)CC1CN(C(=O)Cc2ccsn2)C1 84299,Cc1cc(NC(=O)N(CC(c2ccccc2)(C)C)C)cc2n[nH]cc12 84300,C1(C(=O)NCC(C)OC(F)F)CCCCN1C(C1CCCCO1)=O 84301,C1(NC(C=C(CC)CC)=O)C2CC3CN(C(c4ccc(F)c(N)c4)=O)C1C3C2 84302,c1(C(=O)NC(C2CCCCC2)CNC(C2CCC(O)C2)=O)cn2ncccc2n1 84303,C(CSC)(CC1CCC1)NC(CC)C 84304,C1(C)(CNC(CC(C)C)=O)CN(Cc2cccc(CO)c2)CCO1 84305,c1(C(CC)C(=O)N(C)CCN(C)C(C2CNC(=O)C2)=O)cccc(Cl)c1 84306,c1(C(N(C)CCC2CC2)=O)cc(CNC(C2C3CCC(F)C23)=O)nn1C 84307,CCC(CC1CCCC1)C(=O)N(C)CCN(C)C(C1CC(C)(F)C1)=O 84308,C(=O)(C1=CC(C)(C)C1)NCC(c1ccc(F)cc1F)NC(C(CC=C)OC)=O 84309,c1(C(N2CC(CNC(C(C=C)OC)=O)C(OCC)C2)=O)cccc2ccoc12 84310,C1(C(=O)NCc2ncccc2C)(CC)CCCN(C(c2cnn(C3CC3)c2)=O)C1 84311,N1(C(c2scc(C(=O)OC)n2)C(=O)NC2CC2)CCC(F)(F)C(C)C1 84312,c1(CCC(=O)Nc2oc3ccc(C(C)C)cc3n2)nc(O)c2cc(Br)ccc2n1 84313,c1(NC(C)=O)cnccc1C(=O)NC1C=CCN(C(=O)CS(=O)(=O)NC(C)(C)C)C1 84314,CN1C(=O)CCC1CC(=O)NC1CC2C(NC(C3CCCC(O)C3)=O)C2C1 84315,C1(CNC(c2cc(OC)ncn2)=O)CC2(CC(NC(=O)C(F)(F)CC3CC3)C2)C1 84316,C1(NC(CC(C(=O)O)NC)=O)CCC2(C1)CN(C(c1cc3cn[nH]c3cn1)=O)C2 84317,N1(C(CC=CC=C)=O)CC2CCC2(CCNC(=O)CCc2csc(=N)[nH]2)C1 84318,N1(C(=O)CC2CC2)CCC2(CCCN(C(c3cccnn3)=O)C2)C1 84319,CC1CCC(C)(CNC(c2c(CNC(=O)C(O)C3CC3)nnn2C)=O)CC1 84320,C1(C(NOCC#C)=O)C2CN(C(=O)C(CO)OC)CC12 84321,N1(C(Cc2ccc(OCC)cc2)=O)CCN(C(=O)CNC2CCSC2)CC1CO 84322,c1(CC(=O)NCC(C(C)C)NC(c2cc(F)c[nH]2)=O)cccc(OCC#N)c1 84323,C(=O)(CCCCCNC(=O)CC1CCOC1(C)C)NC(CC(=O)OC)(C)C 84324,C1(C(N2CCC(O)(C(C)NC(C(CC)SC)=O)CC2)=O)CCc2cnc(C)n2C1 84325,C(=O)(CC(CC)C(F)F)N(C1CC(C(N2C(CCC)C=CC2)=O)C1)CC 84326,C(=O)(CCCCC(C)(C)C)N1C2CC(C(=O)NC(c3ccn(C)n3)C)(OC2)C1 84327,C(=O)(CCCCCCBr)N1CCC(C(C(=O)N(CC(=O)NC)C)C)CC1 84328,C(CC(C)CCNC(c1cnn(C(C)CC)c1C)=O)NC(C=C(CC)C)=O 84329,C=CCC(C)(C(=O)NC1CN(C(=O)CC2CCN(C)C2=O)CC1C)N(C)C 84330,c1(C(N2C(C(N3C(C)CCCC3)=O)C3CCC2C3)=O)ccc(S(N)(=O)=O)cc1 84331,c1(C(N(CCOCCNC(C(Br)=C(C)C)=O)C)=O)nc(C)oc1C 84332,C1(NC(=O)Cc2ccc(Cl)s2)CCCC(C(N2CCC(Br)C2)=O)C1 84333,c1(OC)cccc(SCC(=O)NC2CCCC2NC(=O)CN2CC(C)(OC)C2)c1 84334,c1(C(N2C(CO)CC(NC(C(C=C)O)=O)C2)=O)ccc2c(c1C)CCC2 84335,c1(C(N2CC3C(C(=O)Nc4onc(C)c4C#N)(C3)C2)=O)cccc([N+](=O)[O-])c1I 84336,Cc1cc(C)nc(C(=O)NCC2(C(C)(C)O)CN(C(C3CN(C)CC3C)=O)C2)n1 84337,c1(C(=O)NCC2C(NC(=O)Cn3nccc3-c3ccccc3)C2)ccc(F)cn1 84338,C1(CNC(C(CC)(C)CC)=O)CC12CCN(C(=O)CS(=O)(=O)N(C)C)CC2 84339,Cc1cc(Cl)cnc1OCC(N1CCCC1c1cn(-c2ncc(Cl)cn2)nn1)=O 84340,CC(C)C(CNC(c1nnnn1CC1CC1)c1cncs1)C(C)C 84341,C1(C(C)(C)NC(C(N2CCC(OCC)CC2)=O)=O)CCc2ccccc2O1 84342,N1(C(C(C=C)OC)=O)CCC(C(N2CC3(C2)CN(C)C3)=O)C1(C)C 84343,N1(C(CC=CC)=O)CCCC1CN(C)C(c1cscc1SC)=O 84344,Cc1ncc(C#N)cc1NC(=O)C(C1(O)CCC1)NC(=O)Cc1ccc[nH]1 84345,CC1C(=O)CCC1CC(=O)OCCSC1CCCO1 84346,C12(C(=O)NCCCC)C(NC(=O)CC3(O)CCOC3)C3CC1C2C3 84347,N1(CCC(=O)NC2CC(C)(NC(C(CSC)C)=O)C2)C(=O)CCC1=O 84348,N1(C(=O)Cn2cncn2)CCN(C(c2n[nH]cc2[N+](=O)[O-])=O)CC1C1CC1 84349,c1(C(=O)NCCC2(CNC(COC(C)=O)=O)CC2)ccc2nnn(O)c2c1 84350,CS(=O)(=O)CC(=O)N1CCCC1CCCNC(c1cncn1C1CC1)=O 84351,CCC(O)C(F)(F)C(=O)NC1CCN(C(c2cscc2C(F)F)=O)C1 84352,c1(C(=O)NCC(CNC(c2ccc(C3C(C)C3)o2)=O)F)cc(Cl)nnc1O 84353,c1(C(=O)NC2C(NC(=O)Cc3cn[nH]c3)CCCC2)cnc(O)c2ccccc12 84354,C(=O)(C1=CC2CCCCCC12)NCC1(O)CC2N(C(C3CN(C)C3)=O)C(CC2)C1 84355,c1(COC)nc(NCC2(CN(C)C)CCOC2)cc(=NC2CC3(COCCO3)C2)[nH]1 84356,C12CCC(=O)N(C1)C2.C1(COC(C(N)=O)=O)CCCN1C(c1ccccc1)=O 84357,c1(SC)c(NC(c2csc(-c3cc(C)nn3C)n2)=O)cccc1F 84358,Cc1ccc(-c2c[nH]cc2C(=O)NCC2CC2NC(C2CC(N(C)C)C2)=O)s1 84359,C1(C(N(C)CC2CCCN2C(=O)CC(O)c2ccccc2)=O)CC2OC1C1CC21 84360,C1(C(=O)NCC2CC(F)(CNC(c3ccc(F)cc3O)=O)C2)COC2(CCC2)C1 84361,c1(NC)cnncc1C(=O)N(CC(=O)NCC(C)(C)C1(O)CCC1)C1CC1 84362,c1(CC(=O)NCCC2CCN(C(c3cnc(C)s3)=O)CC2)cc(F)c(N)cc1F 84363,CCC(C)CC(C(=O)N1CCC12CC(O)C2)NC(C1CCC(O)CN1C)=O 84364,CN1CCC(NC(=O)CCN(C(c2ncc(F)cc2F)=O)C2CC2)C(C#N)C1 84365,c1(CC)nc(C(C(=O)NC(c2ccccc2)C)N(c2ccccc2)CC)n[nH]1 84366,c1(C(N2CCC(CC(=O)NCCC(COC)O)CC2)=O)cccc2ccoc12 84367,N1(c2c(OC)cncc2)CCCC(C)(C(=O)NCC2CCC(O)C2)C1 84368,c1(C(=O)NCCN(C(=O)CC2OCCCC2(C)C)CC)cc2occc2s1 84369,Cc1cc(C(=O)NC2CN(C(c3csc(C)c3)=O)CCC2CO)nc(C)c1 84370,CCCCCS(=O)(=O)CC(=O)N1CC2CCN(C(=O)Cc3ccccc3)CC2C1 84371,Cc1cc(=NCCCCNC(=O)C(C)Cc2ccccc2C)[nH]c(Cl)n1 84372,c1(CN(c2nc(C)cc(C)n2)C)ccc2c(cnn2C)c1.C12CN(C1)C2=O 84373,N1(C(C(C)n2cccn2)=O)CCOC2(CCCCC2NC(C2CCCN2)=O)C1 84374,c1(CN(C)C)cccc(NC(=O)NC2CCCC2C(F)(F)F)c1 84375,C1(NC(Cc2cc(C)on2)=O)C2CCC1N(C(=O)COCc1nccn1C)C2 84376,c1(CC(=O)OCc2cc(C(C)(C)C)cc(F)c2)cccc2ocnc12 84377,C(=O)(C(C(C)(C)C)OC)N1CC(NC(CC(CC)SC)=O)(CO)C1 84378,N12CC(C(C)C1)C2.c12ccc(cc1)OC2.C(C(O)CO)N(CC)CC1CC1(F)F 84379,CC(CC(=O)NCC1CC1C(=O)NC(C)(C)C(C)(C)C)CC(C)(C)C 84380,c1(CC)cccc(CC(N2CC(NC(C3(CO)CC3(F)F)=O)CC2CO)=O)c1 84381,N1(Cc2cccc(C)c2)CC(C)C(O)C(C)C1.c12nnc(s1)C2 84382,Cn1cnc(C=CC(=O)NC2CCCC2NC(C2(N(C)C)CCC2)=O)c1 84383,C(=O)(CCC(=O)NN(C)C)N1CCC(C)C(CNC(C2CCCCC2)=O)C1 84384,C(C1=NOC2CN(C(c3cccc(F)c3F)=O)CC12)NC(C1CN(C2CC2)C1)=O 84385,C1(C(N(CC(CNC(c2c(SC)ccs2)=O)(C)C)C)=O)CC2CCC1O2 84386,c1(CC(N2CC(CNC(CCCOC(C)=O)=O)C2)=O)ccc2c[nH]nc2c1 84387,C(=O)(Nn1nnc2c1CCCC2)C1(C)CCN(C(CC2CC(OCC)C2)=O)C1 84388,C(=O)(C(C)(C)C(C)C)NC(CC)CN(C(=O)CSc1nc[nH]n1)C 84389,CCC(F)(F)CC(=O)NCC1CC(C)CCN1C(=O)CC(c1ccc(F)cc1)C 84390,N1(C(c2c(OC)scc2)=O)CCCC2(CCCCC2NC(=O)CC2CC2)C1 84391,c1(CC)ccc(C(=O)NCC2(NC(c3cc(F)cnc3O)=O)CCCC2)cc1F 84392,c1(C(N2CCC(N(C(c3c(O)ncc(CC)c3)=O)C)C2)=O)nc[nH]c2ncnc1-2 84393,N1(CC(N2CCC(C(C(=O)NC(COC)(C)COC)F)C2)=O)CCC(=O)CC1 84394,c1(C(=O)NC2CCN(Cc3c(OC)cccc3Cl)CC2O)nc(C)c(C)nc1C 84395,CC1CCC(C(=O)NC2(C(=O)NCC3CCCS3)CCC2)CC1 84396,CCC(CC)(CN=c1[nH]nc(C(C)C)o1)NC(c1nocc1C)=O 84397,CCC(CNC(C1C2CN(C(=O)C(C)(C)C#N)CC12)=O)CC(C)C 84398,N1(C(CCOC2CN(C(COCCOC)=O)C2)=O)CC(O)C(O)C12CCC2 84399,Cc1ccc2c(c1)CC(C(=O)NC(CNC(c1ccc(C(F)F)cc1)=O)CO)S2 84400,CCCCC(F)C(=O)NC1(C(=O)N(C)CC2(O)CCC2)CCN(C)C1 84401,N1(C(C(COC)O)=O)CCC2(C(N3CC(c4ccccc4)C(O)C3)=O)CC2C1 84402,N1(C(C2C(OC)(OC)CC2)=O)CCC2CCC(NC(=O)CC3(CO)CCC3)C1C2 84403,N1(C(c2c(Cl)cn(CCC)n2)=O)CCN(C(c2ccccc2)=O)CC(CO)C1 84404,CC1CN(C(c2ccc(F)cc2Br)=O)CCCN1C(C1CC(C)(C)C1)=O 84405,c1(SCC(=O)N(c2ccc(C(=O)O)nc2)C)ccc2c(c1)OCCO2 84406,Cc1ncn(C)c1C(N1CCOCC1CCNC(=O)CC1CCCC1)=O 84407,N1(C(c2c(C)cnn2C)=O)CCC2CCC(C1)N2C(=O)CCC1CC(F)(F)C1 84408,Cc1cc(C(C)Nc2ccc(-c3nnc(C(C)C)o3)cc2)c(C)o1 84409,C(=O)(C(CCOC)NC(C1CCC2CC12)=O)NCC#CC 84410,c1(OC)cccc(COC(N2CCCC(CN(CC(C)C(C)C)C(C)C)C2)=O)c1 84411,C1(O)(C(N2C(C)CC(NC(=O)Cn3cc[n+](C)c3)CC2)=O)CCCC(C)(C)C1 84412,C(=O)(CC(C(C)C)NC(c1cnc(Cl)n1C)=O)NCC(C(=O)OC)(F)F 84413,CC1(C)OCCC1C(=O)NCC1CCN(C(c2cnc(S)[nH]2)=O)C1 84414,N1(C(CC(=C)Br)=O)CCN(C(=O)Cc2ccc(F)cc2)C2CCCCC12 84415,c1(C2(OC)CC2)cccc(C(N2CC(N(C(=O)C(=O)Nc3ncc[nH]3)C)C2)=O)c1 84416,C1(C(=O)NCCC2OCC(C)(C)C2)CC12CCN(C(=O)Cn1ccnc1O)CC2 84417,C(c1c(F)cccc1F)=CC(=O)N(C)CC1(O)CCN(C(COCC#C)=O)C1 84418,C(=O)(C(C)(C(F)F)NC(=O)OC(C)(C)C)NCCCCN(C(C(CC=C)C)=O)C 84419,C1(NC(=O)Cn2ccccc2=O)CC(NC(=O)C(F)F)C12CCC2 84420,C(=O)(C#CC1CCOC1)N(CC(CN(C(c1c(F)ccc(C(C)C)c1)=O)C)O)C 84421,c1(CNC(=O)CC2C3CN(C(=O)C(c4cccnc4)O)CC23)cnc2n1CCC2 84422,CCC(C)(CO)C(=O)NCc1ccccc1CNC(c1ncn(C)n1)=O 84423,Cc1cc(NC(C2CCCCCCC2)=O)ccc1NC(c1ccncc1O)=O 84424,c1(CC(=O)NCC(n2cc(Br)cn2)C)ccon1.C(C)(C)(C)OC=O 84425,C12(NC(CSc3c(C)cccc3)=O)CCCC1CN(C(=O)C(F)CC1CCC1)C2 84426,c1(C(=O)OCC2C(C)(C)CCCO2)cc(C#N)ccn1 84427,C1(NC(CCC=C)=O)CCN(C(c2ccc(-c3cc[nH]n3)cc2)=O)CCC1(F)F 84428,C(=O)(C(F)(CNC(C1CCCCO1)=O)C(C)C)NCc1n(CCC)ccn1 84429,N1(C(c2c(CCC)occ2)=O)CCCC(CCNC(c2snc(Cl)c2Cl)=O)C1 84430,N1(C(c2c(CC)n(C)nn2)=O)CC(OC)CC1(C)CNC(=O)CSC 84431,c1(C2(C)C(C(=O)NC(C3CCCN(c4nnc(CO)s4)C3)C)C2)ccc(F)cc1 84432,CCCC(F)C(=O)NCCC1(NC(=O)C=CCOCCOC)CCC1 84433,c1(OC)ccc(F)cc1C(N1CCCCC1CNC(=O)C(c1csc(C)n1)=O)=O 84434,N1(CC(N2CC(C)(NC(c3c(C)n(C4CC4)nc3)=O)C2)=O)CCC(=O)NC1=O 84435,C1(C(=O)NCc2c(CC)c[nH]n2)CCCN1NC(=O)C=CC(=O)OC 84436,c1(C(C)=O)ccc(C(c2c(CCC(N3C(C(=O)O)CC3)=O)cccc2)O)cc1 84437,C(=O)(C(F)(F)C(F)F)NCC1N(C(C2(C(F)(F)F)CCCCC2)=O)CCCCC1 84438,C=CC(F)(F)C(=O)NC(CN(C)C(c1cnn(C2CCCCC2)c1)=O)CC 84439,C12(C(=O)NC3CC(NC(C(C)OCCCC)=O)C3)CCCN(CCC1)C2 84440,c1(OC)nc(Br)ccc1C(F)(F)F.C12(OC)CN(C1)C(=O)N2.C12CC(C1)CN2C 84441,C1(NC(CN(CCC)C)=O)CC(C(=O)Nc2cc(C)ccc2CO)C12CCC2 84442,C1(NC(c2nc(CCC)oc2)=O)(CNC(C2C3COCC23)=O)CCCCC1 84443,c1(C(=O)NCCC(=O)NC2C(CN(CC)CC)C2)sc(-c2ccc(C)o2)nc1C 84444,N1(C(C2C(C)(C)C2C#N)=O)CC2(C=C(C(=O)NC3CN4CCC3CC4)CO2)C1 84445,Cc1ncc(NC(N2CCC(Cc3ccccc3)C2)=O)cc1CC(C)C 84446,C1(CC(N2C3C(CNC(c4cnc5sccn45)=O)C(C3)C2)=O)CC(O)C12CCC2 84447,C12(CNCc3c(C(C)C)n(C)nc3)CCCCC1OCC2 84448,n12nnnc1C1(CCC1S)NCC2(C)SCCC(OC)(OC)OC.CCCC 84449,Cc1nnc2cc(NC3CCCC34CN(C(=O)C(C)(C)OC(C)C)C4)ncn12 84450,CC1(O)CCN(CC(=O)NC2CCCCC2CNC(=O)CNC=O)C1 84451,Cc1cccc(C(N2CC(C(=O)NC(C)(C)CCCF)CCC2C)=O)c1C 84452,c1(OC)c(C(=O)NCC(F)CNC(c2c[nH]nc2[N+](=O)[O-])=O)cccc1F 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84541,c1(C(C)C)c(C(=O)NC(C)(CNC(=O)CCC#N)C2CC2)cnc2ncnn12 84542,C(C(CC(F)(F)F)NC(c1nnc(O)cc1O)=O)NC(CC1CCCC(C)O1)=O 84543,S(=O)(=O)(c1csc(NC(c2c(-c3ccc(OC)cc3)nc(CC3CC3)s2)=O)n1)OC 84544,N1(C(Cn2nnc(C)n2)=O)CCOCC(NC(c2cc(NC3CC3)ncn2)=O)C1 84545,c1(C(=O)NCC(CNC(COC2(C)CCC2)=O)CO)ccc([N+](=O)[O-])s1 84546,N1(C(CCC#C)=O)CCCC(O)(CNC(C23CC(CN2C2CC2)C3)=O)C1 84547,c1(C(=O)NC23CC(NC(c4ccon4)=O)(C2)C3)ccc2nccnc2c1 84548,C12(NC(c3c(OC)oc(C)n3)=O)CCCC1CN(C(c1ccc(C)c(C)c1)=O)C2 84549,c1(C(N2CCN(C(C3C(=C)C3)=O)C3C2COC3)=O)cc(OC)cc2c1CCCC2 84550,c1(C(N(C2CCN(C(=O)Cc3nc(C4CC4)nn3C)C2)C)=O)ccc(CF)cc1 84551,c1(C(=O)NCC(C)(O)C(F)F)[nH]nc2ncccc12 84552,Cc1noc2cc(N3CCN(C4CN(C)C5(CCC5)C4)CC3)nc(Cl)c12 84553,C(=O)(C1=CNC2=NCCC2=C1)NC1(C)CCN(C(C(COCC)(C)C)=O)C1 84554,S(=O)(=O)(CCCCCl)N(c1ccc(NC(=O)NCCCO)cn1)CCCO 84555,C1(C(N(CCCNC(C2C(C)C2C)=O)C)=O)CC12CC(F)(F)C2 84556,C(CC(=O)NOCC(C)(C)C)OC(CNC(C(C1CCCC1)OC)=O)(C)C 84557,CCC(C)CC(=O)NC1CC1NC(=O)OC(C)(C)C.C12CC(C1)NC2=O 84558,C1(C(=O)NCC2(CNC(C(CC#C)C)=O)CCCCC2)COc2ccccc2C1 84559,C1(C(N(C(C)C(N2CCOC(C3CC3)CC2)=O)CC)=O)CCC=CCCC1 84560,N1(C(C2C(=C)C2)=O)CCN(C(c2ccc(-n3cncn3)c(N)c2)=O)CC(C)(F)C1 84561,C1(NC(C2C=CC(NC(C(C)n3cccc3)=O)C2)=O)CCCC2(CC1)CC2 84562,c1(C(N2CC(NC(C34CCC(CC3)OC4)=O)CC(O)C2)=O)ccc2nncn2c1 84563,CCCCCC(O)C(C)C(=O)N1CCC=C(CNC(=O)CC2CCCCO2)C1 84564,c1(CC(=O)OC)ccc(S(=O)(=O)NC(c2occ(C)c2C)=O)cc1 84565,C1(NC(C(C)OCCC=C)=O)CCCC1NC(c1cc(CC(C)C)on1)=O 84566,C1(N2CCC(COC)C2)C(C)OCC12CCN(C(c1cc(Br)ccc1Br)=O)CC2 84567,C(=O)(C(C(C)C)OCC(C)C)NCC(CC)NC(c1sncc1C)=O 84568,N1(C(C(CCC)NC(N)=O)=O)CC(C(N2CCC(O)C(CO)C2)=O)CC(C)(C)C1 84569,N1(C(C(C)OCC)=O)CCN(C(c2cccc(OCC(F)(F)F)n2)=O)CC1C 84570,C(=O)(C1SCCc2sccc21)N1CCC(N(C(=O)C(O)CC(F)F)CC)CC1 84571,C(=O)(C(CC)C(F)(F)F)NCC(CCCC)NC(=O)C1=CCCC1 84572,CN1CCC(N2CC(C(=O)NCC3(CN(C(=O)CC4(C)CC4)C)CC3)C2)CC1 84573,C(=O)(C(C)(C)C(C)C)NCC1CC(NC(c2c(C(=O)OC)c(C)[nH]n2)=O)C1 84574,CC1CCN(C(c2cc(CNC(=O)NCC(C)NC(c3ccco3)=O)cs2)=O)C1 84575,CCC(C(=O)NC1(CCCNC(=O)CCCN2CCCCC2)CC1)C(C)C 84576,c1(C(=O)NCC(CC=C)NC(=O)CN2CC3CC3C2)cnn(CCO)c1C 84577,C1(COC)CN(C(C23CC(NC(=O)CC4CC4C4CC4)(C2)C3)=O)CCO1 84578,C(=O)(C1=C(Cl)CCOC1)N1CCC(O)(C(C)NC(=O)C(F)(F)c2ccccn2)C1 84579,c1(C(=O)OCC)ccc(S(=O)(=O)NCC(O)C(N)=O)c(Br)c1 84580,N1(C(C2(CC)CCC2)=O)CC(N(C)C(c2cc(OC)cnn2)=O)C2(CC2)C1 84581,C1(NC(c2cc(C)no2)=O)COCCC1NC(=O)CCc1cc(Br)cs1 84582,Cc1onc(Cl)c1C(=O)N(CCCNC(c1c(C(F)(F)F)n[nH]c1C)=O)C 84583,N1(C(c2ccc([N+](=O)[O-])[nH]2)=O)CC2(CCC(C(N3CCC(F)C3)=O)O2)C1 84584,C(c1ccc(Cl)cc1Cl)=CC(=O)N(CCCCCCNC(C(CC)(C)CO)=O)C 84585,N1(C(CCSCCCC)=O)CCC2CN(C(=O)C(C3CCC3)OC)CC12 84586,N1(C(CCOC)=O)CCCC2(CCN(Cc3cc(C(N)=O)n[nH]3)C2)C1 84587,C1(CNC(=O)C=CCF)CCCN(C(=O)CNS(=O)(=O)C2CC2)CC1 84588,c1(N2CCN(C(C=C(C)C(=O)O)=O)C(C(F)(F)F)C2)ncnc2[nH]c(C)nc12 84589,N1(C(C2OCOC(C)C2C)=O)Cc2ccc(CNC(=O)CCC3CC3)cc2C1 84590,c1(NC(C2C(NC(CC=C)=O)CCCC2)=O)ccc(C)c(CC)c1 84591,c1(OC)ccc(NC(c2nc(-c3c(SC)cccc3F)sc2C)=O)cc1OC 84592,c1(NC(C2CCOC2)CNC(c2ccc(OC)nc2)=O)c([N+](=O)[O-])cnn1C 84593,Cc1ccc(C(=O)NCC(C)NC(c2c(C)noc2N)=O)cc1[N+](=O)[O-] 84594,Cc1cc(Br)cc(S(=O)(=O)N2CC3(CCC(NC(c4nccs4)=O)C3)C2)c1 84595,N1(C(c2c(C)ncnc2C)=O)CCN(C(c2cc3ccccc3s2)=O)CC(O)C1 84596,C12(C)CCCN(C1)CCC(=O)NC(=O)C(CC)N2.C(=O)(NC)NC1CC1 84597,C(=O)(C1=CC2CCC(C1)C2)NCCN(C(=O)CC1C(C)(C)C1(C)C)C 84598,C1(C(=O)NCC=CCSC)CC12CCN(C(=O)C(C)C(=O)OC)CC2 84599,Cc1ccc(C23CC2CN(C(=O)NCCc2noc(C)n2)C3)cc1 84600,Cc1cncnc1C(=O)NC1(CNC(=O)COc2cccc(F)n2)CC(F)(F)C1 84601,C1(CNC(=O)NC(CC=C)CC)CCC2(CC1)CC2(F)F 84602,Cc1cccc(F)c1CC(=O)NC1C2CC1CN(C(=O)CC1COCC(C)O1)C2 84603,c1(C(N2CC(N(C(=O)Cc3ccns3)C)C2)=O)cc(Cl)cn1C 84604,N1(CC)CC(NC(=O)C(CN(C)C)NC(c2cccs2)=O)CC1=O 84605,c1(NCCN2CCN(C(C3CCC(CSC)C3)=O)CC2)ncc([N+](=O)[O-])c(C)n1 84606,CC1=C(C(=O)N(C(C)CNC(c2nn(C)c(C)c2Br)=O)C)SCCO1 84607,NS(=O)(=O)c1cccc(C(=O)NCCNC(=O)CCSCc2ccccc2)c1 84608,Cc1cc(F)sc1C(=O)NC1(CNC(c2cc(C(F)(F)F)[nH]c2C)=O)CCCC1 84609,C(=O)(CC1C(=O)Nc2cc(Cl)ccc21)NCC1(NC(C)=O)CCOC1.C1C(=O)N1 84610,C=CCC(CC=C)C(=O)NC1CN(C(=O)Cn2cnc(=N)[nH]2)C2CCCC12 84611,CC(C)C1=NOC(C(=O)N(CC(=O)NCC2CCC(=O)O2)C)C1 84612,CN=c1[nH]cc(C(=O)NCC2CCC(NC(c3cnc[nH]3)=O)C2)o1 84613,c1(CN(C(C(C)NS(C)(=O)=O)=O)CCNC(=O)CCN2CCCC2)ccccc1 84614,c1(CN2C(CCC(=O)NC(C(=O)OC)C3CC3)CCC2)ccc(C#N)s1 84615,c1(CCC(=O)OCC)ccc(N2CCCC2C2(NC(=O)C(C)(C)F)CC2)nc1 84616,c1(COCC(=O)NCCN(C)C(C2CN(C3CCCCC3)C2)=O)ccncc1 84617,c1(COC)cc(C(=O)NCC2C(C)CCN2C(c2ccc[nH]2)=O)c(C)o1 84618,C1(CC)CCN(C(=O)C(CC)N(C)C)C1CNC(c1ncncc1Cl)=O 84619,C1(C(=O)NCC2(CSC)CC2)C(C2CC2)CCN1C(c1cnccc1C#N)=O 84620,C12(C(=O)NCCCCCNC(C3CC34CCOC4)=O)CCN(CC1)CC2 84621,N1(C(C(CC)C2CCOCC2)=O)Cc2nccn2CC(NC(=O)C(F)(F)CO)C1 84622,CC1(CNC(c2cc(F)c[nH]2)=O)CCN(C(=O)CN2CCCC2CO)CC1 84623,C1(C(C)NC(c2c(CC)cns2)=O)CCCN(C(c2n[nH]cc2Cl)=O)C1 84624,C(c1c(F)cccc1F)=CC(=O)N(C)CC1(NC(C2C=CCCC2)=O)CC1 84625,C=CC(C)CC(=O)NC1COCC1NC(=O)C(C)=C1CC1 84626,N1(C(CSSC)=O)CC2(CCC(CNC(=O)CNC(=O)CCC(C)C)O2)C1 84627,N1(C(C2CC(N(C)C)C2)=O)CC(O)CC1(C)C(=O)NC(CO)C(F)(F)F 84628,C#CCC(C)(C)C(=O)NCC1CCN(C(=O)CCOCCOC)C12CC2 84629,C1(C(=O)NC2CCN(C(Cn3nc(C)c(Br)c3)=O)C2)CCC2C(C1)C2(F)F 84630,CCC(C)CCCCC(=O)N1CC(NC(=O)C=Cc2cnccn2)C2(CCC2)C1 84631,C(=O)(C1c2ccccc2CN1C(c1cnc(C)c(C)c1)=O)NCC(=O)NC 84632,c1(C(=O)OCC(=O)Nc2cccc(CNC(C=CC)=O)c2)nnc2ccccn12 84633,C(=O)(CCCCC(F)(F)F)N1CCC(N(C(=O)C(C)C2CC2)CCOC)CC1 84634,C1(C(=O)NC2CCCC2NC(c2cccnc2O)=O)(OC)CCCC(C)(C)CC1 84635,C(C1c2ccccc2CN1C(C1C2COCC12)=O)NC(C(NOC)=O)=O 84636,N1(C(Cc2c(C)ccs2)=O)CC2CC(NC(C3CCC(C)(C)O3)=O)CC1C2 84637,N1(C(C(CC=CCC)C)=O)CCC(N=[N+]=[N-])(C(=O)NC2(CCC)CC2)C1 84638,Cc1cc(C(=O)N(C(C)(C)CC(=O)NC2CCCC2(C)O)C)nc(O)c1 84639,C1(C(=O)NCC2(C(C)NC(Cc3c(C)ocn3)=O)CC2)CC2C=CC1CC2 84640,C1(O)(CC(=O)N(CCCOCCNC(C2(CC=C)CC=CC2)=O)C)CCCCC1 84641,N1(C(c2c(OC)c(C)ccc2)=O)Cc2ccnn2CC(NC(=O)CCCC#N)C1 84642,c1(C(N(C2CCN(C(=O)COCc3nnc[nH]3)C2)CC)=O)cccc2sncc12 84643,c1(CC)ccc(F)cc1C.C1N=C(NC(C)C)NCC2(CCC2)ON2CCCC12 84644,N1(C(c2cc(SC)oc2)=O)CC2CCCC2C1C(=O)Nc1cccc(Cl)c1 84645,C=CCC(C)(C)C(=O)N1C2CCC(C2)C1C(=O)NC1CONC1=O 84646,c1(OC2(C(=O)NC3C(CNC(c4c(C)cns4)=O)C3)CC2)ccc(Cl)cc1 84647,C1(NC(c2cc(C)[nH]n2)=O)CCC2CC1CN2C(=O)C(O)C(C)C 84648,C1(CNC(c2c(CNC(c3cnc(SC)s3)=O)ocn2)=O)CN2CCC1C2 84649,N1(C(C=CC(C)C)=O)CCC2CCN(C(c3ccc(F)c(C(F)F)n3)=O)CC2C1 84650,c1(SCCN2C(C(F)(F)F)CNCC2)c(Cl)c[nH]c2nccc1-2 84651,N1(C(C2CN(C(CSCC)=O)CC2C)=O)CCC(C2CC2)C1 84652,C(CC(C)(C)C(=O)NCC(CO)NC(C1(F)CCN(C(C)(C)C)C1)=O)OC 84653,c1(C(N(CCCCNC(CC(CC)OC)=O)C)=O)cc2cccc(Cl)c2[nH]1 84654,c1(C(=O)NCc2ccc(C(C)NC(COCC)=O)cc2)nnn2c1CCCC2 84655,C(=O)(C(C)C1=CCCC1)N1CC(COC)(NC(=O)C(c2ccc(C)cc2)(F)F)C1 84656,N1(C(C2(NC(C3C(OC)(OC)CC3)=O)CC(F)C2)=O)CC2CCCC(O)C2C1 84657,C(=O)(CCN=[N+]=[N-])N(CCC(=O)NC(c1nc(=O)o[nH]1)C)CC1CC1 84658,CC(N=c1[nH]c2c(c(=NCc3ccn(C)n3)[nH]1)CCCC2)c1ccc(O)nc1 84659,C1(N(C(=O)C(F)C2CCCC2)C(=O)CC2CCC2)CCC2CCC12 84660,Cc1cc(C(N2CC(NC(c3cc(C4CCC4)nn3C)=O)C2)=O)ncc1C(N)=O 84661,C1(C(N(CC#CC)C)=O)CC2(CC2)CN1C(C1CC12CCC2)=O 84662,c1(C(=O)Nc2c(C)cc(NC(C3CCCOC3)=O)cc2)ccnc2c1cnn2C 84663,C1(C(C(=O)NC(C)C)N(CC(C)C)Cc2ccnn2C)CCCOCC1 84664,C(C(C(=O)NCCc1cn(C)cn1)NC(=O)Cn1cccn1)OC 84665,C1(C(=O)NC2(CN(C(=O)Cc3ccc(F)cc3)C)CC2)Cc2cc(Cl)ccc2O1 84666,S(=O)(=O)(c1cc(Br)c(C)cc1F)N1CCCC(CN(CCC)C)C1 84667,Cc1ccc2c(C(=O)NCCC(C)NC(=O)C(C)C(C)(C)C)coc2c1 84668,N1(C(C(CCOC)C)=O)CC2(CCCC2NC(=O)CC2(OC)CCOCC2)C1 84669,N1(C(c2c(C)nc(Br)s2)=O)CCC2C(CCN2C(c2cc(Cl)cc(Cl)c2Cl)=O)C1 84670,CCCC(CCC)C(=O)NC1CN(C(=O)Cc2cc[nH]n2)C1 84671,C1(N(C(c2cnc(CCCC)[nH]2)=O)C)CCCCN(C(c2cc(C#N)no2)=O)C1 84672,C(C(C(C)(C)C)NC(C1(C)CC1(Cl)Cl)=O)NC(C(C)c1cncs1)=O 84673,C1(NC(c2ccc(OC(F)F)cn2)=O)C2CC1CN(C(=O)C=C1CCC1)C2 84674,N1(C(c2c(C#C)c[nH]n2)=O)CCC2(CC1)CCN(C(=O)CCCC(F)F)CC2C 84675,C1(NC(CCOCC)=O)CC(C)(NC(c2cnc[nH]2)=O)C1 84676,C1(Nc2ncccn2)CCCCN(C(=O)CCOCC(=O)NCC2CCCO2)C1 84677,N1(C(C(CC)(C)C)=O)CCC(O)(CCNC(c2cc(C)c(C)nn2)=O)CC1 84678,C1(CC(C(=O)NC2CC2)N(CCC)Cc2ccc(O)cc2)CCOC(C)(C)C1 84679,C12(CNC(=O)CCN3CCC3)CC(C1)C(NC(=O)C1=COCCO1)CO2 84680,c1(CC)cc(=NC(=O)CC2CN(C(=O)CC(O)C(C)C)CC2C)[nH]n1C 84681,N1(C(c2n(C)c(S)nn2)=O)CC(CNC(=O)C(=O)NC2CC2)CC12CCC2 84682,Cc1cccnc1CC(=O)NC1CCN(C(=O)Cc2ccc(Cl)cc2)CC1 84683,c1(C(=O)NCC(CC)NC(=O)CCCCCSC)c(C)cccc1O 84684,C1(NC(C2CCN(c3n(C)ccn3)C2)=O)COCCC1NC(=O)Cc1cn[nH]c1 84685,C1(CCC)CN(C(=O)C(C2(O)CN(C(C3(C4CC4)CC3)=O)C2)F)CCO1 84686,C(C(C)CC(=O)N(C(C)C(C)(C)O)C)NC(c1c(C)nco1)=O 84687,C1(C(N2CC(CNC(=O)C(F)(F)CC3CCCO3)C2)=O)CCc2[nH]nc(O)c2C1 84688,Cc1nc(CC(=O)NC(c2cccnc2)C(=O)NCCCC(=O)N(C)C)cs1 84689,CC1CC(C)N(C(c2coc(CO)c2)=O)CCN1C(=O)CC1CN(C)C1 84690,C(=O)(C(O)CC(F)(F)F)N(C1CCN(C(c2ccc(O)nc2Cl)=O)C1)CC1CC1 84691,Cc1nc(CC(F)(F)F)sc1CC(=O)NCCN(C(=O)C(O)CF)C(C)C 84692,C1(C)(CNC(c2cn(C)nc2C(F)F)c2n(C(C)C)nnn2)CC2CC2C1 84693,C12(NC(C(C)=C3CC3)=O)CCCC1N(C(c1cnn3c1OCC3)=O)CCC2 84694,C12(NC(CCC)=O)CC1CN(C(c1cnn(Cc3ccccc3)c1F)=O)C2 84695,C1(NC(CC(CCC)(C)O)=O)CCC2CCN(C(c3cc(C)nn3C)=O)C1C2 84696,C1(OC)(CN)CCN(C(=O)C(=Cc2cccnc2)N=[N+]=[N-])C1 84697,CC(C)CN(CC(O)C1CC1)C(C)C 84698,C1(CNC(C(C)OCCN(C)C)=O)CN(C(C2C3CC4C(C3=O)C24)=O)CC12CC2 84699,N1(C(C(C)Cn2ccnc2)=O)Cc2cccn2CC(C(N2CCOCC2)=O)C1 84700,CC1CC(CNC(=O)CCOCC(F)F)CN1C(=O)CCN1CCCC1=O 84701,C1(C(=O)NC2C(NC(=O)CCc3ccc(F)cc3F)CC2)Cc2ccccc2C1 84702,C12(NC(c3cn(CC(N)=O)nn3)=O)CCCC1(F)CN(C(C1CCC1)=O)C2 84703,CC1CC2(CC(C(=O)NOCC(=O)NC3(C(F)F)CCC3)C2)C1 84704,n1(CC(=O)N(C(CNC(COCCSC)=O)C)C)ccc(=O)c([N+](=O)[O-])c1 84705,C1(NC(CC(C=C)(C)O)=O)CCCCCN(C(=O)CS(=O)(=O)C2CC2)C1 84706,N1(C(C(CC)OCC)=O)CCN(C(=O)C=Cc2c(C)coc2C)C(CC)C1 84707,c1(NC(C(c2csc(Cl)c2)N(CC)CC2CCOC2)=O)ccc(F)cc1 84708,c1(OCC)oc(C)nc1C(=O)NC1CC(N(C(=O)CC(O)c2ccccc2)C)C1 84709,C(C(F)(F)C(=O)NC1CCOCC1C(=O)NCCC(C)(O)C1CC1)OC 84710,C12CCCCCN1C2=O.C1(CC(=O)NCCOCCOCCSCC)CC(F)(F)C1 84711,c1(N2CCCC(C)(CNC(CC3CC(C)C3)=O)C2)ccc([N+](=O)[O-])cc1C(C)=O 84712,Cc1nn(CC(=O)NCCN(CCOCCO)C(C2(O)CC(F)(F)C2)=O)c(=O)o1 84713,C1(NC(c2cccc(C)c2)=O)CC2CCC(C1)N2C(C1(CF)CC2(CCC2)C1)=O 84714,c1(CN2C3CN(C(C4N(C)CCC4)=O)C(C3)C2)ccc(F)c([N+](=O)[O-])c1 84715,C1(C)(CNC(C2C(C)C2)=O)CCN(C(C2CC23CC(O)C3)=O)C1 84716,C1(C(N(C2CCCN(C(C(c3ccn(C)n3)C)=O)C2)CC)=O)CCCC(C)(C)C1 84717,c1(C(N2CC3C(C(=O)NCCCC(=O)OC)(CC3)C2)=O)c(F)cc(Br)cc1Br 84718,c1(CC(=O)NC2(CNC(C(COC)C)=O)CCCCC2)c(F)cccc1F 84719,C(CC(=O)NC1CCC(c2nncn2C)CC1)(C(F)(F)F)OCC 84720,C1(NC(c2ccn(CC(C)C)n2)=O)(CO)CCCN(c2ccc(C#N)nc2)C1 84721,Cc1ccc(C(c2nnnn2C)NC(c2cccc(F)c2C)C)cc1Cl 84722,CC1(C)CCCC(CC(=O)NCC2(C)CCCC2NC(=O)Cn2cccn2)C1 84723,N1(CCC(=O)NCCOC(CNC(C(C)SC)=O)(C)C)CCNC(=O)C1 84724,C(=O)(CCCC(F)(F)F)N1CC(C)C(C)(C(=O)NC2CCn3ccnc3C2)C1 84725,C1(NCCN(C(CC)C)CC)CCC(C)(C)C1.C(C)(C)(C)OC=O 84726,c1(C(=O)NC(c2ccc(F)cc2)CC)cc(C)c2sccc2c1 84727,C1(NC(C2C(=C)C2)=O)CC(C)CN(C(c2ccc(-n3cccc3)cc2C)=O)C1 84728,N1(C(c2nc(OCC)oc2)=O)CCC(NC(C2CC(=O)N2)=O)C(C)(C)C1 84729,C1(NC(c2ccnc(OC)n2)=O)CC2CC1CC2C(=O)NCCC(F)(F)F 84730,c1(NC(N2CCC(n3cc(C4CC4)nn3)C(O)C2)=O)cc(F)ccc1Br 84731,C(Cn1cncn1)(C(=O)NC1C2CCCC12)NC(C1CC(=C)C1)=O 84732,c1(OC)cc(C)cc(C)c1C(C)NC(c1ccc(C)c(C)n1)c1nnnn1C(C)C 84733,N1(C(c2c(CC)onc2C)=O)CCC(NC(=O)C=CC2CCCC2)C(C)C1 84734,c1(C(=O)Nc2ncc(C)c(I)c2)n[nH]c2c1CCN(C(c1ccc(O)cn1)=O)C2 84735,C=CCC(C)(O)C(=O)NC1C2CC3C1C3C2C(N1CCN(C)C(CC)C1)=O 84736,C1(C2N(C(C3(CC=C)CCC3)=O)CCC2)CCN(C(=O)CC(C)CC)CC1 84737,C=CC1OCCC1C(=O)NCC(c1ccc(F)cc1)NC(c1csnc1OC)=O 84738,C1(C(=O)NCCCCCN(C)C)CCN(C(C2(C)C=CCCC2)=O)CCO1 84739,C1(N(C(c2ccn(CC)n2)=O)C)C2CN(C(C3(O)CCOCC3)=O)CC12 84740,C(=O)(C1=NOC2(CCOC2)C1)N1CCCN(C(C2C(=O)NCC2)=O)CCC1 84741,CCCC(C(=O)NCC(C)(C)C(=O)NCC1OCCC1C)N(C)C 84742,C(CN=C(NCC1CC2(C1)CC21CCC1)N1CCC(C(C)(C)C)CC1)OCC 84743,c1(N(C(=O)C(C)OC2CCCC2)CCN(CC)CC)ncc([N+](=O)[O-])c(C)n1 84744,C#Cc1cc(F)cnc1NC(C1CN(C(c2cncc(F)c2)=O)CCC1O)=O 84745,N1(C(c2c(OC)nsc2OC)=O)CCC(C)C(NC(C2SCCCS2)=O)C1 84746,C1(CNC(C(COC)C)=O)CN(C(c2ccc(F)s2)=O)CCC12CCC2 84747,c1(C(=O)NCCC(C)N(C(=O)CC2(C)CCCCC2)C)cc(Br)cn1C 84748,CCC(C)CC(=O)NCC1(NC(=O)CSCC(N2CCOCC2)=O)CCCC1 84749,C1(F)(C(N(CCCCC=C)C)=O)CCN(C(C2SCC=C2C)=O)CC1 84750,Cc1cc(-c2nc(C3CCC3)nn2-c2cccc(Br)c2)c(C)[nH]1 84751,C(=O)(C1=NOC2(CCOC2)C1)N1CC(F)(CNC(=O)Cc2cncs2)C1 84752,C1(NC(CN(C2CCCC2)C)=O)CCN(C(=O)CSc2nncs2)CC1 84753,C1(C2CCN(C)CC2)(C(N2C(CNC(COCCOCC)=O)CCCC2)=O)CC1 84754,N1(C(c2ccc(N)c(F)c2)=O)CC2(CCCC2NC(C2CCCC23CC3)=O)C1 84755,Cc1c(NCC(C2CCCC2)N(C)C)ncnc1N(C)CCc1ccco1 84756,N1(C(c2ccc(NC=O)cc2)=O)CC2CC1CN2C(c1cnc(C2CC2)o1)=O 84757,c1(C(N2CC(CC(=O)N(C)Cc3ccccc3Cl)OCC2)=O)cnc(O)cc1O 84758,c1(C(C(=O)N(CC(C)N(C)C(c2sccc2F)=O)C)C)ccc(Cl)s1 84759,c1(C(=O)NCC2(O)CN(C(C3CCC4CC34)=O)C2)c(F)cccc1[N+](=O)[O-] 84760,C1(C(=O)NC(C(C)NC(c2cc(C(F)(F)F)cs2)=O)(C)C)CCCN(CCF)C1 84761,C1(C(C)C)C(NC(C2CC2c2cccs2)=O)CCN1C(=O)COc1cccnc1 84762,CC1CN(C(c2ccoc2)=O)CC2(CCN(C(c3cccc(N)c3O)=O)CC2)O1 84763,C1(NC(CCOCCN(C)C)=O)CC(O)CN(C(c2ccc(O)nc2Cl)=O)C1 84764,C(=O)(C(CO)C(F)(F)F)N(CC(C)O)CCNC(=O)C=CC1(C)CCOCC1 84765,c1(CC)nc(N2CCC(C(C)NC(C3CCN(C(C)=O)CC3)=O)C2)[nH]c(=N)n1 84766,Cc1cc(C(=O)NCCNC(C2CCCN2C(N)=O)=O)c2c(C)noc2n1 84767,CN1C2CCC1CC(C(N1CC3(CCC3NC(c3cccn(C)c3=O)=O)C1)=O)C2 84768,CC1CN2CCN1CC2NC(c1ccccc1OC(C)(C)C)=O 84769,S(=O)(=O)(c1cn(C)nc1C)N1C(C(=O)Nc2c(C)ccc(Cl)c2)CC(O)CC1 84770,C(=O)(C(C)(C)C1CCCN1Cc1ccncc1)N(C1CC(=O)C1C(F)(F)F)C 84771,CC(CN(C)C)CCC(=O)NC1C=CC(NC(=O)COCC2CCOCC2)C1 84772,c1(C(N2CCN(CC)CC2C)C(=O)NCCC#N)nc(Cl)cc(C)c1Br 84773,c1(CN2CCC(c3cccc(C(=O)NC4CCC4)c3)CC2)cc(Cl)cc(Br)c1F 84774,C(=O)(CC1OCCc2ccccc21)NC(CNC(C1(OC(C)C)CCC1)=O)(C)C 84775,C(CCC(C)C)(C(=O)Nc1cn(C)nc1C)NC(CN(C(=O)OC)C)=O 84776,c1(SC)cc(C(=O)NC2CCC2NC(=O)C(c2cncn2C)O)ccn1 84777,CCC(C)CCCCC(=O)NS(=O)(=O)c1ccc(C#N)o1 84778,c1(OC(C(=O)NCC(C)NC(=O)CC(O)c2ccccc2)C)ccc(CO)cc1 84779,c1(NC(C)=O)ccc(C(=O)OCc2cnn(C)c2Br)cc1 84780,C1(C(N2C(CNC(c3n(C=C)ncc3)=O)CCCC2)=O)CCc2nnc(O)n2C1 84781,CC1(CCNC(C2(n3nccn3)CC2)=O)CCN(C(C2CCCC(=O)O2)=O)C1 84782,c1(NCCNC(C2CCCN(C(CSCC#C)=O)C2)=O)cnc(CC)nc1C 84783,C1(C(N(CC#C)CCO)=O)N(C(=O)C(C)CSC)CCC1(C)C 84784,Cc1ccc(F)cc1NC(=O)CN1CCC(NC(=O)C(C)n2cccn2)C(O)C1 84785,C(=O)(C1=NOC(C)(C)C1)NC1CCCC(NC(c2c(C)ncc(C)c2)=O)CC1 84786,C1(NC(C(C)(C)NC(Cc2cn(C)nc2)=O)=O)CC12CC(O)C2 84787,C(=O)(CCCC(=O)N(c1ncnc(C)c1Br)C1CCNCC1F)OC 84788,C#CCC(C)(C)C(=O)NC(C1CCCN(C(c2cc(C)nn2CC)=O)C1)C 84789,Cc1cc(C(=O)N(C2CN(C(=O)C(CC(C)C)NC(N)=O)C2)C)ncc1C#N 84790,NS(=O)(=O)c1ccc(CC(N2CCCC23CCN(C(C2CC(F)C2)=O)C3)=O)cc1 84791,N1(C(CCN(CCC)C)=O)CC(c2ccccc2)(NC(c2occc2F)=O)C1 84792,C1(NC(C(C)Oc2cccc(Br)c2)=O)CCN(C(=O)C=CCO)CC12CCC2 84793,c1(C(=O)NCc2cn(-c3cc(C)c(Cl)nc3)nn2)c(Br)cc(F)c(F)c1F 84794,c1(CN(C)C(C2(CNC(C34CCC(C3)C4)=O)CC2)=O)ccn(C)c1 84795,c1(C(N2CC(C)(CC(=O)Nc3ccc(Cl)cc3)C2)=O)cc2cc(Br)ccc2s1 84796,C(=O)(CCCCC(=O)NC1CN(C(C2(O)CCOC2)=O)CC2(CC2)C1)NC 84797,C1(NC(=O)CCCn2cncn2)CCOC1(C)C.c12nocc1C(=O)NC2C 84798,C(C(C)(C(=O)NCC(CO)NC(C1(CCc2ccccc2)CC1)=O)OC)OC 84799,n1(CC)nc(C)c(C(N2CC3CC2C3CNC(C23CCOC(C)(C2)C3)=O)=O)c1Cl 84800,N1(CCn2c(C)cc(-c3ccccc3)n2)CCC(O)C(C)C1 84801,Cc1cc(C(=O)NC2(C)CC(NC(C3CC(=O)NC(C)C3)=O)C2)cc(C)n1 84802,CON1CC(C(=O)NCCCN2CCC(NC(C3CC4C=CC3C4)=O)C2)CC1=O 84803,N1(C(C2CC(OC)C2)=O)CCC2(CC2)CC1C(=O)NC(CCO)C1CCC1 84804,CC1OCCC1(F)C(=O)NCC1CCCN(c2ncnc(C(C)(C)C)n2)C1 84805,C1(CNC(c2ccc(CCC)[nH]2)=O)CN(C(=O)CN2CCCC2)CCC12CCC2 84806,c1(NC(C2NCCN(C(c3c(C)ncnc3)=O)C2)=O)ncnc2[nH]c(Br)nc12 84807,N1(C(c2c(CC)occ2)=O)CC(NC(C2CC(C#N)C2)=O)CCC1C 84808,CC1CCOC1CCNC(=O)C(C1(C)CC1)NC(=O)Cc1ccon1 84809,C1(C(=O)NCc2cccnc2Br)CC12CCN(C(c1cn[nH]c1)=O)C2 84810,c1(C(CC)C)ccc(C(=O)NC2(C)CN(C(c3occc3C)=O)C2)cc1 84811,C1(C(=O)NC2CC(C(C)C)C2)CCN(C(C2(CC3CC3)CC2)=O)CCO1 84812,C1(NC(CC(C)C)=O)CC2CC(NC(C3CNC(=O)N3)=O)CC12 84813,S(=O)(=O)(c1cccc(=NCC(C)C(C)C)[nH]1)N1CCC(CCCOC)CC1 84814,N1(N(C(=O)CCC2CC(NC(c3ccc(C(C)=O)o3)=O)C2)C)CCC(CC)C1 84815,c1(C2(C(=O)NCC(C)(O)CNC(c3csc(Cl)n3)=O)CC2)cccnc1Cl 84816,C1(CNC(=O)C(N2CCCC2c2ccc(Cl)cc2)=O)CCCS(=O)(=O)C1 84817,C1(=CCNC(C=CCCC(C)C)=O)CCN(C(c2c(C(C)C)cnn2C)=O)CC1 84818,C(=O)(C(F)CC(CC)CC)NC1(C(=O)NCCNC(CC)=O)CCOCC1 84819,CC1(CS(=O)(=O)Nc2ccc(Cl)cc2)CCCN(CC(N2CCCC(CO)C2)=O)C1 84820,N1(C(c2cnn(C(C)(C)C)c2)C(=O)NC(C)C)Cc2ccccc2C(C)(C)C1 84821,CC1CSCC1(c1nnnn1C(C)(C)C)NCCOc1ncccc1Br 84822,c1(C(C(=O)NCC#CCNC(C2OCCN(C)C2)=O)=O)ccc(F)cc1F 84823,C1(NC(CNC(N)=O)=O)CCOCC1NC(c1cnc(Cl)[nH]1)=O 84824,Cc1cc(C)c(N(C(c2cccnn2)C2CNC2=O)CC2CCCO2)c(C)c1 84825,C(=O)(NNc1ccc(Br)c(F)c1F)NCCC1(C(=O)OCC)CCOCC1 84826,C1(C(=O)NCCOCCOCC)CCOCC1NC(=O)C=NOC 84827,CC1CN2CCN1C(C(=O)NC1C=CCN(C(c3cnc4[nH]ccc4n3)=O)C1)C2 84828,C1(c2cn(Cc3c(C)nc(CC)o3)nn2)CN(C(c2ccnn2C)=O)CC1(C)C 84829,C(C(C)(O)CC(=O)N1CCC1CNC(=O)C(C)(C)Nc1ccc(Cl)cc1)OC 84830,N1(CC(CC)CC(C)(C)C)CC(C(=O)OC)C2(CN(C(=O)OC(C)(C)C)C2)C1 84831,N1(C(C2(O)CCCCC2)CC)CCN(C(C2C(NC(=O)C(C)(C)OC)C2)=O)CC1 84832,C1(NC(CCC)=O)CC(C)(C(=O)NCC(CO)C2CCC2)C1 84833,n1(CC(=O)NCC(CNC(C23CCCC(CO2)C3)=O)CO)cnc2ccccc12 84834,C1(C(N2CC(CCNC(C=CC(CC)C)=O)OCCC2)=O)CC(C)(C)C(C)(C)C1 84835,C1(C(=O)NOCc2cccnc2)CCCC1NC(c1ccoc1)=O 84836,FC1CC2CC1CC2NCc1cccc(C2CC2)c1 84837,N1(C(=O)CC2CCCC2(F)F)CC2CCCC(C1)N2C(c1cncc(Cl)c1)=O 84838,c1(C(=O)NC(C)CCNC(c2cc(Br)co2)=O)n[nH]cc1[N+](=O)[O-] 84839,c1(C(=O)NCC2CC(F)(CNC(CCN(C)CC)=O)C2)sc(C#N)cc1Cl 84840,Cn1cc(C(=O)NC2C3CC2N(C(=O)Cc2ccc(C#N)nc2)C3)ccc1=O 84841,C#CCCCCCC(=O)N1CC2CCC1CN2C(=O)CCCC 84842,N1(CC)CC(C(=O)NCCC(C)(C)NC(C2CC(=O)N(O)C2)=O)c2ccccc21 84843,c1(C2OCCN(C(=O)Nc3nnc(NC(=O)C4CC4)s3)C2)ccc(F)c(F)c1 84844,N1(C(c2n(CC)cc(Cl)c2)=O)CCCC(N(CC(N2CCC(C)CC2)=O)C)CC1 84845,c1(C(=O)NCCNC(CC2C(C)C2)=O)cccc2c1NC(=O)CC2 84846,c1(C(=O)NCC2CCN(C(=O)C#CC3CC3)C23CCC3)ccnc2nccnc12 84847,N1(C(c2c(C)cno2)=O)CCC2(CCCN2C(c2ccc(C(C)C)c(Cl)c2)=O)C1 84848,C1(F)(CNC(c2ccoc2)=O)COCCN(C(=O)Cc2ccc(Br)cn2)C1 84849,C1(SCC)CC(C(=O)NCC(C)(C)CCNC(c2nc(O)sc2C)=O)CCO1 84850,c1(C(N2CCN(C(C(C)=C3CC3)=O)CC2C2CC2)=O)cc2cc(Br)ccc2[nH]1 84851,N1(C2CCN(C(CSCC(N)=O)=O)CC2)CCN(C(=O)CO)CC1=O 84852,CC(=O)CCCC(=O)N1CCC(C)C1CNC(=O)C(O)C1CCC1 84853,C1(NC(c2c(OCC)ccs2)=O)CS(=O)(=O)CC1NC(c1c(Cl)cnn1C)=O 84854,c1(CNCC2N(C(c3c(OC)cncc3)=O)CCOC2)cc(F)ccc1Br 84855,N1(CC(C)(C)O)CCN(C(CC2CCCC2)C(=O)NCCc2ccccn2)CC1 84856,CS(=O)(=O)C1CC(C(=O)NCC2CCN(C(=O)CC3COC(=O)C3)C2)C1 84857,C1(CNC(c2c(CC)non2)=O)CCN(C(c2cc(OC)cc(C)c2)=O)CC1C 84858,C(=O)(C1CC(=O)c2c(F)cccc21)NCC(CNC(c1c(C)cccc1Cl)=O)C 84859,c12c(NC)cccc1NC(=O)CCNC2c1n(CC=C)nnn1.C1(CN(C)C)CC1 84860,C1(NC(C(C(C)C)C)=O)CC(N=c2ccn3nccc3[nH]2)C1(C)C 84861,N1(C(C2N(C)CCOC2)=O)CC2(C)CN(C(C3CC(F)(CO)C3)=O)CC2(C)C1 84862,N1(CC)CC2CN(C(=O)C(C3CCCN(C(=O)COCOC)C3)C)CC2C1 84863,c1(C(N2CC(OC)C(NC(C3(C)CC=CCO3)=O)C2)=O)cc(Cl)cc2c1CCC2 84864,C(=O)(C=CS(C)=O)NCCN(C(CN(C(=O)OCC)C)=O)Cc1ccccc1 84865,c1(C(N2CC(C)C(C)C2)=O)ccc(O)c(-c2ccccc2)c1 84866,C1(NC(c2c(CC)n(C)nn2)=O)CC(CNC(=O)CCc2cnn[nH]2)C12CCC2 84867,C(=O)(C(CNC(=O)C1=CCCC1C)C(C)C)NC(COC)(C)C(N)=O 84868,CN1CCn2ncc(C(=O)NC3(C)CCCN(C(=O)COCC(C)(C)C)C3)c21 84869,N1(C(c2ccc(C)cc2F)=O)CCCC(C2CCN(C(c3nncs3)=O)C2)C1 84870,C1(C(N2CC(C3CN(C(C45CCC(CC4)CO5)=O)C3)C2)=O)CCc2cnnn2C1 84871,Cc1ccc(C(N2CCC(NC(=O)CC3CCC(C)(C)C3)CC2)=O)c(O)c1 84872,CC1CC=C(C(=O)NC2(C(=O)NCC3(CO)CCC3)CSC2)CC1 84873,c1(NC(=O)NC2(C(=O)NC3CC3NC(=O)CC3CSC3)CC2)ccccc1 84874,CN1CCCC(CCC(N2CCC(C)(NC(=O)Cc3nc[nH]n3)C2)=O)C1 84875,c1(C(=O)NC2CC(NC(c3cc(C)c(Br)s3)=O)C2)cccc(Br)c1O 84876,N1(C(C(Cc2c(C)nc[nH]2)O)=O)CCC(NC(=O)CCCCCN(C)C)C12CC2 84877,O=C(C1=CSCCO1)NCC(c1ccccc1)CNC(C1CCCO1)=O 84878,N1(C(c2c(C(C)C)cco2)=O)CC(NC(c2ccc(Cl)s2)=O)C2(CCOCC2)C1 84879,N1(C(C(C(C)C)F)=O)CCCC(F)(CNC(=O)C=CC2CC2)CC1 84880,c1(CC)ncccc1NC(=O)CC1CCCN1C(c1cncc(Br)c1)=O 84881,c1(C(=O)NCC2CCN(C(CC(n3ccc(C)n3)C)=O)C2)cccnc1C 84882,CC1=C(C(=O)N(C2CC(NC(c3ccnc(OC(F)F)c3)=O)C2)CC)SCCO1 84883,C1(CNC(C(C(C)C)N(C)C)=O)CN(C)CCN1C(c1csnc1Br)=O 84884,c1(C(c2nnnn2CCCF)Nc2ccccc2COC)cc(Cl)ccc1[N+](=O)[O-] 84885,C(CC(=O)N(C1CC2CC2C1)C)(C(C)CC)NC(c1cn(CC=C)nn1)=O 84886,c1(NC(C)=O)cccc(C2CCN(C(C3CCN(c4ccccc4)C3)=O)C2)c1 84887,c1(C(=O)NC2CCN(CCNC(CC(C=C)C)=O)CC2)c(F)ccc2n[nH]cc12 84888,C1(C(C)C)CN(C(C2CC(=O)C2C)=O)CCN1C(C1CS(=O)(=O)C1)=O 84889,C(=O)(C(C)(C)C(=O)N1CCC(C(CO)NC(=O)C(C)c2cc[nH]n2)CC1)OCC 84890,c1(C(N(CC=CC(N2C(C(C)O)COCC2)=O)C)=O)coc2ccccc12 84891,c1(C(=O)NCC(CC=C)NC(=O)C(C)(F)CCCC)cnc2c(ccn2C)c1 84892,N1(CCC(N2CCC(NC(C3CCC(C#C)CC3)=O)C2)=O)Cc2ccccc2C1 84893,c1(CC)ccc(C(=O)N(C(C)CNC(c2cnn(C)c2Cl)=O)CC)c(F)c1 84894,N1(C(C2(C=C)CC2)=O)CCC2(CCC2NC(c2ccc(C)nc2)=O)CC1 84895,C=CC1(C(=O)NCCCCCN(C(=O)Cc2csc(NC=O)n2)C)CCC1 84896,C1(NC(Cc2c(C)noc2)=O)CCCC(NC(=O)C(C)C=Cc2ccccc2)C1 84897,C1(C)(C(=O)NC2CCC(C(=O)NC(CCC)c3ccco3)C2)CCC(=O)N1 84898,C1(C(N(C(C)C)C)=O)CC2CC2N1C(C1(F)CC1(Cl)Cl)=O 84899,c1(CNC(C(C)N(C(C2C(CC)C2)=O)C)=O)ccnn1C 84900,c1(C(=O)NC2CC(NC(c3ncnc4sccc34)=O)C2)ccc2cc[nH]c2c1 84901,c1(C(C(=O)NCCC)N(CC)Cc2ccc(OC)cc2)ccc2c(c1)CC(C)O2 84902,c1(C(N(CC(CC)NC(C23CCC(F)C2CC3)=O)CC)=O)nc(O)nc(O)c1F 84903,C1(C)(NC(C2C(C)OCC2)=O)CCCN(C(c2c[nH]cc2Br)=O)C1 84904,C(N=c1[nH]c2c(c(=NC3CCOC(C)(C)C3)[nH]1)CCC2)c1ccc(C)c(N)c1 84905,Cc1ccc(C)c(C(=O)NC(C)CN2CCN(C(C3(C)CC(C)C3)=O)CC2)c1C 84906,N1(C(C2CCC(=O)NC2)=O)CCN(C(=O)Cc2cc(Cl)ccc2Cl)C(CCO)C1 84907,Cc1cc(C(=O)NC2COCC2NC(=O)C#CC(C)C)c(C)cc1Br 84908,C1(NC(=O)CC2(O)CCOC2)CN(C(C2CCN(CCF)CC2)=O)CC12CCC2 84909,c1(C(=O)NCC(N(C(c2cc(C)ncn2)=O)C)C2CC2)ccc(Cl)cc1O 84910,c1(C(=O)OC)cncc(OCCNc2ccsc2Cl)c1 84911,CC1CC(NC(c2cnc(Cl)n2C)=O)CCN1C(c1cc(F)cc(Cl)c1)=O 84912,C1(CNC(c2ccc(CSC)o2)=O)CCCCC1NC(=O)CCc1n[nH]c(=N)s1 84913,C1(NC(=O)C2=CCC2)COC2(CCCN(C(c3cc[nH]c3C3CC3)=O)C2)C1 84914,c1(C(N2C(C(C)NC(C(CCSC)N(C)C)=O)CCC2)=O)cnc2sccc2c1 84915,C1(c2n(CCCSCC)nnn2)(OC)CCCC1CNCC(c1nncn1C)(C)C 84916,C1(C(N2CCC(N(C(C3C(=C)C3)=O)CC)C2)=O)CC2(C1)CS(=O)(=O)C2 84917,CCC(C)C(C(=O)N1CC(C(=O)NC2CCN(OC)CC2)C(F)C1)N(C)C 84918,C1(NC(CCC=CC)=O)CN(C(C2(F)CCCC2)=O)CCC1CO 84919,N1(C(c2ccn(C)c2-c2ccccc2)=O)CC(S(N)(=O)=O)C1 84920,N1(C(C2CC(NC(c3ncc(C)[n+]([O-])c3)=O)C2)=O)CC2CC3CC2C1C3 84921,C1(c2cn(CC)nn2)CN(CC(F)(F)C(F)F)CCC1(F)F.Cc1cc(C=O)no1 84922,Cc1cn2c(n1)CC(C(=O)NC1CCN(C(=O)COCCO)CC1CO)CC2 84923,c1(OC)cc(OC2CC2)ccc1C(=O)NC1CC(CNC(=O)CC2CCCO2)C1 84924,C1(CNC(CCC#N)=O)CCCN(C(C2CCC(CN3CCOCC3)O2)=O)C1 84925,N(C1COc2ccccc21)C(=O)CCn1cc(Cn2cccc2)nn1 84926,c1(CC(N2CCC(=CC=C)CC2)=O)ccc(-c2ccccc2)c(F)c1 84927,CCCC(C(=O)N(C)CC1CC(O)C1)NC(c1cn(C)cc1C)=O 84928,C1(OC)(CNC(c2nnnn2C2CCOC2)CCc2ccccc2)CCCCC1 84929,n1(CCC)cccc1C(=O)N(CCO)Cc1ccn(CC)n1 84930,C=CCC(C)(CC)C(=O)N1CCC(N2CCN(C)CC2)C(C)C1 84931,C1(N(C(C)C)C(c2c(CCN3CCCCC3)cccc2)(C)C)CC12CCNCC2 84932,C1(S(C)(=O)=O)(C(=O)NC(CNC(C(CC)(C)OC)=O)C)CCOCC1 84933,c1(C(=O)NCCC(C)NC(=O)C(C)(F)F)cc(Br)cc2ccccc12 84934,N1(C(c2cncc(C)c2)=O)CCN(C(C2(F)CCS(=O)(=O)C2)=O)CC1CC1CC1 84935,N1(C(c2cnn(-c3ccccc3)c2F)=O)CCCN(C(C2(F)CCOC2)=O)CC1 84936,C(=O)(C1=CCCC1C)NCCN(CCC)C(C1CC1c1cnc[nH]1)=O 84937,C1(OCCC(N2CC(CC(C)NC(C=C(CC)CC)=O)C2)=O)CCOCC1 84938,c1(C(=O)NCCC(C)NC(c2c(SCC)cccc2)=O)ccc2oncc2c1 84939,N1(C(C2CN(C(=O)NC)C2)=O)CC(C)(C)OC2(C1)CN(C(=O)Cc1cnoc1)C2 84940,C=CCCCCC(C(=O)NCCC)N(C1CCN(S(C)(=O)=O)CC1)C 84941,c1(CC(=O)NCC(C2CC2)NC(C(C)(O)C2CC2)=O)ccc2c(c1)OCCCO2 84942,C1(CC)(NC(=O)C(c2nc(C)cs2)C)CCN(C(C2CN(C(=O)N(C)C)C2)=O)C1 84943,C1(C(=O)OC)CCCCCN1C(=O)CN1CCCNS1(=O)=O 84944,NC(=O)CCCC(=O)NC12CC(CNC(=O)CC3CC(O)C34CCC4)(C1)C2 84945,CCC(CNC(c1ccccc1)=O)(CC)NC(=O)CCNC(=O)C(C)O 84946,c1(N(CCC(N)=O)C)nc(=NCCCCCO)[nH]c2c1SCC2 84947,C(C(CC(F)(F)F)NC(C1(c2cc[nH]n2)CCC1)=O)NC(=O)Cc1cn[nH]c1 84948,C(C)(CC(C)NC(c1cc(F)n[nH]1)=O)NC(C=C(C)C(F)F)=O 84949,c1(C(N2C3C(CNC(c4cc(OC)no4)=O)C(C3)C2)=O)cc2n(n1)C(C)CCC2 84950,C(=O)(C#CC1CCOCC1)N1C(C(N2CC(C=C)C2)=O)CN(C)CC1 84951,C1(OC)CN(C(c2ccc(O)nn2)=O)C(C)(CNC(c2ccnc(S)c2)=O)C1 84952,C(=O)(C1=CCN(C(=O)CC23CCCC2C3)CC1)NCCN(C(CC)C)C 84953,c1(OC)cnc(F)c(C(=O)NC2CCCC(NC(c3cccc(C)n3)=O)CC2)c1 84954,N1(C(C=CCCC)=O)CCOC2(CCN(c3nc(O)c4ccccc4n3)C2)C1 84955,N1(C(C2C(C)=C2)=O)CCC(C2CCN(C(c3cccnc3N)=O)CC2)CC1 84956,c1(C(=O)NC2C(C)N(C(=O)CC3CC3)CCC2C)cc2c(F)ccc(Cl)c2[nH]1 84957,C1(NC(c2cnc(C)nc2)=O)C(C)(C)C(NC(=O)CC2CC2C2CC2)C1(C)C 84958,c1(C(N(C)CCOCCNC(C2(CO)CCCC2)=O)=O)c(Cl)cccc1[N+](=O)[O-] 84959,C1(CNC(c2c(OC)csc2)=O)COC(C)(C)CN1C(C12CC(C1)C2)=O 84960,c1(C(=O)NC2CC(CNC(c3c(Cl)nc(OC)s3)=O)C2)cnc(O)cc1C 84961,N1(Cc2ccc(C(N3CCOCC3)=O)[nH]2)CCSC2CCC12 84962,CCCCC(C(=O)NCCC(C)NC(=O)CCOC1CCCC1)NC(N)=O 84963,C(CC(C)(C)C(=O)N1CCN(C(=O)CCCc2ccc(OC)cc2)C(C)C1)OC 84964,c1(C(C)(C)C)cnc(CNc2nccn2CC(F)(F)F)o1 84965,C1(C(=O)NC2CCC(NC(c3cccc(Cl)c3Cl)=O)C2)CCC2CC1CO2 84966,N1(C(CNC(c2[nH]cc(C(=O)OC)c2)=O)C)CCC(CN(C)C)CC1 84967,CC1(C)C(C(=O)NCC(C)(C2CC2)NC(c2cc(F)cc(F)c2)=O)CCS1(=O)=O 84968,C1(C(N(CC(C2CC2)OC)C)=O)CNC(=O)CN1C(=O)Cc1cc(C)ccc1C 84969,Cc1cc(OCC(N2CC(NC(=O)Cn3ncnn3)CCC2C)=O)cc(C)c1 84970,Cc1cc(C(=O)NCC2(CNC(=O)C(C)C3CCCC3)CCCC2)cnn1 84971,C1(NC(Cc2c(C)non2)=O)CCCC2CN(C(c3cn(C)nn3)=O)CC12 84972,C1(C(=O)NC(C2CN(C(=O)CCCC3(C)N=N3)C2)C)CCc2cnn(C)c2C1 84973,Cc1cc([N+](=O)[O-])cc(C(=O)NC2CCN(C(=O)C#CC3CCCC3)C2)c1Cl 84974,C#Cc1ccc(F)c(C(N2CC(C)C(NC(=O)C=C3CCCCC3)C(C)C2)=O)c1 84975,c1(OC)cccc(CNC2CC(C(=O)N(C)C)C2)c1Cl 84976,C1(CC(=O)NC(C)CC(=O)NC2CC2)CCCC(=O)N1.C12(CC1)C(=O)N2 84977,n1(CC)cc(C(=O)C(=O)NCC(C)(C)OCCNC(C2(C)CCCS2)=O)cn1 84978,C1(NCC(c2cn(CC)nc2)O)CCN(c2ccc(Br)cc2)C1=O 84979,C1(C#N)(C(=O)NC2C(C(N(C(C3CCCCC3)C)C)=O)CCC2)CCCCC1 84980,c1(C(=O)OC)nn(C)nc1C(N1CC(CNC(=O)CC2OCCC2C)(OC)C1)=O 84981,CCC(CC(=O)NCC1(C(=O)Nc2cccc(O)c2)CC=CC1)SC 84982,N1(C(C2(C)COC2)=O)CCOCC(F)(CNC(c2cn(C3CCC3O)nn2)=O)C1 84983,C1(CC)CC(N=c2[nH]c(=NC(C)c3ccccn3)[nH]c3c2CCCC3)CCO1 84984,C(CC1CCCO1)(C(=O)NC1CCOC1)N(CC(C)(C)C)CC(C)C 84985,N1(C(c2ccn(CCOC)n2)=O)CCSCC1CCNC(=O)C(C)CC1CCC1 84986,C(=O)(CC1=NNC(=O)C1)N1CC(C(N)=O)(CNC(c2ccc(OCC)cn2)=O)C1 84987,N1(C(CCOC(C)=O)=O)C(C(=O)NCCc2ccco2)C2CC(O)C1C2 84988,C(CCC)(CCCNC(=O)CCc1ncc[nH]1)NC(C(CC=C)NC(C)=O)=O 84989,c1(C(=O)NC(CC)CN(C(=O)CCC(C)C)C)cccc(F)c1C#N 84990,N1(c2snc(C)c2C#N)CCC2(NC(=O)CCCN3CCCC3)CCCCCC12 84991,c1(-c2cc(C(=O)OC(CC)C)n[nH]2)c(C)[nH]c2ccccc12.C12CSCN1C2=O 84992,N1(C(C2(Cl)CC2)=O)CC2CCN(C(C34CC5CC(CC3C5)C4)=O)CC2C1 84993,CCC(CC(=O)N1CCCC1CNC(=O)CC(=O)OC(C)(C)C)CC(C)C 84994,n1(CC(=O)N(CCCN(C)CC2CC2)CC2CCO2)cnc(C(=O)OC(C)(C)C)n1 84995,c1(C(=O)NCCC(=C)CNC(c2oc(Br)nc2C)=O)cn2ccccc2n1 84996,N1(C(CCSCCCC)=O)CCC2(C1)CN(C(C1(C)CCN(C)CC1)=O)CCO2 84997,N1(C(C(C)n2cccn2)=O)CC2CCC(NC(=O)C3=CCN(C)C3)(C2)C1 84998,C1(C(C)C)COCCN(C(C2CCN(C(=O)C(C)(C)C3CC3)CC2C)=O)C1 84999,C1(NC(C(CC)c2ccccc2)=O)CCC(NC(=O)C(C)(C2CC2)OC)CC1 85000,c1(CC)nc(C(=O)NCC2C(CNC(=O)CC(C)OC)C2(F)F)cs1 85001,C1(SC)CCN(C(C2C3CCCC23)C(=O)Nc2cccc(Cl)c2C)C2(CC2)C1 85002,C1(CC(=O)N(C(C(N2CCC(CSC)C2)=O)C2(C)CC2)CCO)CCN(C)CC1 85003,N1(C(CN(C(CCc2c(C)noc2)=O)C2CC2)=O)CCCC1(C)CC(C)C 85004,c1(C(N(CCNC(c2c[nH]nc2Br)=O)CC)=O)nccc(OC)c1N 85005,N1(C(CCOCC)=O)CCC(C2CCN(C(c3ccnc(C4CC4)c3)=O)CC2)C1 85006,c1(C(=O)NCCC(C)NC(c2cn(CCC=C)nn2)=O)c(C)nn2c1NCCC2 85007,C(=O)(C(C)C(O)C(C)C)N(C1CC(C#N)C1)CC(=O)NC(C=C)CO 85008,C(=O)(C(CNC(C1CCCC1O)=O)C(C)(C)C)NCCSC 85009,C1(CC(=O)NC2CCC(NC(C3(C)CCCOC3)=O)CC2)CCC(=O)NC1=O 85010,N1(C(c2c(C)c(O)ccc2)=O)CC(CNC(C2(C)CCN(C)C2)=O)CC(C)(C)C1 85011,c1(-c2nc(C(C)OCC(C)C)n(CCN(C)C)n2)ccc(Cl)c(Cl)c1 85012,C=CCC(CO)NC(=O)C(C)CNC(=O)CCC1CC1C 85013,N1(C(c2c(CC)scc2)=O)CC(C)(C)OCC1CNC(=O)C(c1ccc(C)o1)C 85014,C=CC(CCC)CC(=O)NCCOC1CN(C(c2cn3ccnc3s2)=O)C1 85015,c1(N(CC(C2CCC2)OC)C)nc(N2CCCOCC2)c2c(n1)c(C)nn2C 85016,C1(C(=O)NCC(CC)NC(C2(C)CCCOC2)=O)CCC12CCC2 85017,N1(C(C2N(C)CSC2)=O)CC2(CNC(=O)C(F)C3CCC3)CC1CO2 85018,N1(C(c2cnc(C(C)OC)s2)=O)CCCC(CCNC(c2oncc2C)=O)C1 85019,C1(CC(=O)NCc2nc(CNC(C3CCCN(C)C3)=O)sc2)CCCS(=O)(=O)C1 85020,N1(C(c2csc(C)c2N)=O)CCC(NC(C2CCC(C(N)=O)N2C)=O)CC(O)C1 85021,C1(C(=O)NC2CC(NC(c3c[nH]nc3CNC)=O)C2)COCCN1C1CCCC1 85022,c1(C(N(C)CCNC(c2cnc(C3CCOC3)s2)=O)=O)csc2nnsc12 85023,CCC(C(=O)OCCNC1(C)CC1)n1ccnc1.C12(CC1)C(C)(C)N2 85024,Cc1sc(N)c(C(=O)NCC2CCCC2NC(c2cnn(C)c2C(C)C)=O)c1C 85025,N1(C(c2cccc(CC)c2F)=O)CC2(CCCN(C(c3cccc(C)c3)=O)C2)C1 85026,N1(C(C(C2CCOCC2)OCC)=O)CCN(C(c2ccoc2)=O)C2COCC12 85027,N1(C(CC)=O)CCCC(C2(NC(=O)CCCCCF)CC2)C1 85028,Cc1n[nH]cc1CNC(=O)C=CCC1(NC(=O)CCn2ccnc2)CCC1 85029,C12(CNC(CC=CC)=O)CC1CN(C(C13CC(c4ccccc4)C1C3)=O)C2 85030,c1(OC)ccccc1C(C(C)(C)C)NC(c1ccc(N2CCCC2)cc1)=O 85031,N1(CC(=O)N(C2CCCC2)C)CCC(NCC2CC2)CC1 85032,c1(C(N2C(CNC(C(C)CN(C)C)=O)CC3(CC3)C2)=O)cc2cc(N)ccc2[nH]1 85033,c1(C(N2CC(NC(C(C)O)=O)C(CO)CC2)=O)ccc2occc2c1 85034,Nc1ccc(Cl)c(C(=O)NCC2CC(NC(=O)C3=CCCOC3)C23CCC3)c1 85035,N1(C(c2n(CCC)ncc2)C(=O)NC2CC2)CCCC(O)C1 85036,CC1(C)CCN(C(=O)Cc2cncnc2O)C(C(=O)NC2CCCCC2(C)C)C1 85037,S(=O)(=O)(c1cc(C(N2CC(CC#C)OCC2)=O)ccc1OC)NC(C)=O 85038,c1(-c2nc(C)sc2)cccc(C(N2CC3(NC(C4CCC4)=O)CC2C3)=O)c1 85039,N1(C(C(CO)N(C)C)=O)C2CC=C(C(=O)NC3CCC4(CCCC4)C3)C1CC2 85040,C1(C(N2C(CC(=O)NC)CC2)=O)CN(C(c2cc(O)ccc2C)=O)C(C)(C)C1 85041,C(N=c1cc(C)nc(N2CC(CO)C3(CC3)C2)[nH]1)NCC(C)(OCC)OC 85042,c1(CN(C(CNC=O)=O)CCNC(=O)C(F)(F)c2nccs2)ccc(F)cc1F 85043,N1(C(C2CN(C(C)=O)C2)=O)CCN(C(c2nn(C)cc2C)=O)C2CCCCC2C1 85044,CCN=C(NCc1ccc(NC(C)=O)nc1)NC1CCCC1(F)F 85045,C1(NC(CC(C)CF)=O)CCC2(CCN(C(c3cc[nH]c4nccc3-4)=O)CC2)C1 85046,C1(N(C(CSCC#C)=O)C)CN(C(c2c[nH]nc2C)=O)CC1F 85047,c1(NC(CC)(CCCl)c2nnnn2C2CCCCCC2)cc(Br)ccc1OC 85048,C1(CC)C(=O)NCCN1C(C1CCCN1C(=O)CCCc1cnn[nH]1)=O 85049,CCCC(C)C(=O)NC1CCCC1CNC(c1sc(=N)[nH]c1C1CC1)=O 85050,c1(NC2C3CN(C(c4c(C)nc(C)s4)=O)C(C3)C2)ncnc2c(F)cccc12 85051,C1(NC(C2=CC(C)(CC)C2)=O)CN(C(=O)Cc2csc(C)c2)Cc2ccnn2C1 85052,C1(CCNC(C(C)(C)c2cc[nH]n2)=O)COCCN1C(=O)C=Cc1cccs1 85053,S(=O)(=O)(c1cccc2c1OCCO2)Nc1ccc2c(c1)N(C)CC2 85054,C=CC1OCCC1C(=O)NCC1CC(=O)NC1=O 85055,C(C(C(=O)NCC1(O)CC(N(C)C)C1)NC(=O)C(O)C1CCCC1)OC(C)C 85056,C(C(C)C(=O)NC1CNC1=O)OCC.C(CCSCC)NC(C)=O 85057,Cn1ncc(C(N2CC=C(CNC(C3CC34CCOCC4)=O)CC2)=O)c1C#N 85058,C1(C(CS(C)(=O)=O)NC)CCC(F)(F)CC1.C12CCCN(C1C)C(C(=O)OC)C2 85059,N1(C(=O)OCCC=C)CC2CCC1(C(=O)NCCC(F)(F)F)CC2 85060,Cc1c(O)nnc(N2CCN(c3ncc(Br)cn3)CC2)c1C 85061,N1(C(CNC(=O)Nc2c(CC=C)nn(C)c2)=O)CCN(C(CCCC)=O)C2CC12 85062,c1(CC(N2CC=CC(NC(c3cc(C(C)C)sn3)=O)C2)=O)ccc(F)cc1F 85063,C1(C(N(CC#C)CC)=O)CC2CC1CN(C(C1CCC(=O)CC1)=O)C2 85064,c1(CCOC(CCC2(C)CN(C(=O)OC(C)(C)C)C2)=O)cc2ccccc2s1 85065,N1(C(C=C(CC)CC)=O)CCCCC12CC(NC(=O)C(C)Cc1ccncc1)C2 85066,N1(C(COCCCC)=O)CC2CN(C(=O)C(c3ccccc3F)(C)F)CC2(C)C1 85067,c1(N2CCC(CCOC)(NC(=O)C(C)SC)CC2)ccc([N+](=O)[O-])cc1C#N 85068,N1(C(CCc2onc(SC)n2)=O)CCC2(NC(c3ccnc(C)c3)=O)CCCC12 85069,C1(NC(C(CSC)OC)=O)CC2(C1)CC2C(=O)NCC1COCCN1C 85070,C(=O)(C#CC1(C)CCCO1)NC1C(NC(Cc2n(C(C)C)cnn2)=O)CCCC1 85071,N1(C(C(CNC(c2c(C)nsc2C)=O)OC)=O)CCCC(C2(C)CC2)C1 85072,c1(OC(C)C)ccc(C(=O)NCCC2(NC(C34COCC3C4)=O)CC2)cc1 85073,C1(CNC(CSC(C)C)=O)CCCCCN1C(C1CC1c1cnc[nH]1)=O 85074,Cc1ccnn1CC(=O)NCC(O)C(=O)NC(c1cn[nH]c1)C 85075,N1(C(CC(C(C)C)O)=O)CCN(C(c2ccn(C(C)(C)C)n2)=O)C(C)C1C 85076,CCC(C#N)C(=O)N(C1CCN(C(C2CCN(S(=O)(=O)CC)CC2)=O)C1)CC 85077,c1(C(N2CC(C(C)NC(c3nsnc3O)=O)C2)=O)ccc(-c2cccs2)nc1O 85078,C1(CC(N2CCCC(N(C)C(c3n[nH]cc3F)=O)C2)=O)NC(=O)CNC1=O 85079,C1(C(=O)NCCn2ncc(CC)c2)CN(C)CCN1C(C1CCCC(=O)N1)=O 85080,C1(CNC(CC=CC=C)=O)CCC2CN(C(c3ncc(C=O)s3)=O)CCC2C1 85081,C1(NC(C2C(CC)CCC2)=O)CCC(NC(c2cc(OC)c(Cl)s2)=O)CC1 85082,S(=O)(=O)(c1cccc(F)c1)NCCNC(c1cn(CCOC)nc1)=O 85083,N1(C(=O)CCCCCn2cc(C3CCCOC3)nn2)CCCC2(CCNC2)C1 85084,N1(C(c2cccc(OC)c2OC)=O)CCCCC12CN(C(c1ccoc1C)=O)C2 85085,C1(COC)CN(C(c2cc(F)n(C)n2)=O)CCN1C(c1ccn(C2CC2)c1C)=O 85086,Cn1ccc(C(=O)NC2(C(=O)NC3CC(CO)C34CCC4)CCCCC2)cc1=O 85087,N1(C(C)C(=O)NCC(F)(F)F)CCC2(CN(C(=O)C(C)(C)C3CCCO3)C2)C1 85088,C1(O)(CCNC(C(C)OCC#C)=O)CN(C(=O)Cn2nccn2)C1 85089,CCC(CC(=O)NC1(CC(=O)NCC2CC[Si](C)(C)C2)CC1)C(C)C 85090,Cc1cccc(CC(=O)NC2CCC(CNC(C3(C)CSC3)=O)C2)c1 85091,Cc1ccc(C)n1CC(=O)NC1C=CC(C(=O)NCC2CCC(C)C2)C1 85092,c1(OC)cc(O)c(CN2CCCC2c2ncc(-c3c(F)cccc3Cl)[nH]2)cc1O 85093,C1(C(N2CC(N(C(C(CC)CC)=O)C)C(C)CC2)=O)CCCC2(CCC2)C1 85094,c1(C(N(CC(C)NC(=O)C=CSC)CC)=O)csc(C)c1C 85095,CC(C)(C#N)CCCCNC(=O)NCC1(CC(F)F)CCCO1 85096,C(=O)(C1COc2ccccc21)NC1CCN(C(c2n[nH]c(C)c2C)=O)CC1C 85097,C(=O)(CC1OC(=O)c2ccccc21)NCCCCNC(CCCC(CCC)C)=O 85098,C1(NC(C2(F)CCN(C(C(C)C3CCCO3)=O)CC2)=O)CC2CC1CC21CC1 85099,c1(C(=O)NC(CNC(C(CC)=CC)=O)CC)nccc(C)c1N 85100,N1(C(c2nn(C)c(OC(F)F)c2)=O)CC(NC(=O)CCCn2ccnc2)CC(O)C1 85101,C(C(=O)NCC(C1CC1)N(C)C(c1ccc(SC2CC2)cn1)=O)(C(C)C)NC(C)C 85102,c1(C(N2C(C)CC(NC(=O)CS(N)(=O)=O)CC2)=O)ccc2n[nH]cc2n1 85103,O=C(CC(F)(F)F)N1CC(N2CCN(C(c3c[nH]ccc3=O)=O)CC2)C1 85104,C(=O)(C1=NOC2(CCOC2)C1)NCC1(OC)CN(C(=O)C(F)n2cccn2)C1 85105,N1(C(c2ccc(CC)s2)=O)CCC(O)C(NC(C2(C)CCCCO2)=O)C1 85106,C1(NC(CCOCCCOC)=O)CN(C(=O)C=CSC)C(C)(COC)C1 85107,N1(C(C2C(C)OCC2)=O)CCC(C(C)(C)C)(CNC(=O)COC(F)(F)F)C1 85108,N1(C(c2ncccc2Cl)=O)CCC2(CCCC2Nc2nccc(CO)n2)CC1 85109,c1(C(=O)NC(CNC(C2(C(=O)OCC)CC2)=O)C)ccc(N)cc1C 85110,C1(CNC(C(C)(C)CO)=O)COCC2(CCN(C(=O)CC3=CCCCC3)C2)O1 85111,CC1CN(C(C2CCC(n3cc(-c4c[nH]nc4F)nn3)C2)=O)CC1CO 85112,C1(C)(CC)C=C(C(=O)NC2CCCC(NC(c3nnn(C(C)(C)C)n3)=O)C2)C1 85113,N1(C(c2occ(C)c2)=O)CC(C)CN(C(=O)OC(C)(C)C)c2ccccc21 85114,N1(C(c2c(O)ccc(C)c2)=O)CC2(C1)SCCC2NC(=O)C1=CC2CCCC12 85115,N1(C(c2c(C)ncnc2O)=O)CC(O)(C2(CNC(=O)C3=CCCC3)CC2)C1 85116,C1(NC(CC2OCCC(C)(C)C2)=O)CC2CCC(C1)N2C(=O)CC1C=CCC1 85117,C12(NC(COCCCCC)=O)CC(C(=O)NCC3(F)CC3)(C1)C2 85118,C1(O)(CN(C(c2ncn(CC)c2)=O)C)CCN(C(c2ccoc2Cl)=O)C1 85119,C=C(C)CC(C(=O)NC1CCN(C(=O)CC2(COC)CC2)C(C)C1)OC 85120,C12(CNC(CNc3[nH]c(=N)sc3)=O)CNCCN1CCOC2 85121,C(=O)(CS(=O)(=O)CCO)NCC(CCNC(c1cc(CC)ncc1)=O)O 85122,N12CCC3CCN(CC13)C2=O.c1(OCCOCC#C)cc(F)c(C)cc1C#N 85123,C1(OC)(OC)CC2(CN(CC3CC(C4CC4)=NO3)C2C(=O)O)C1 85124,N1(C(C(CC=CCC)C)=O)CC(C)N(C(=O)CSC(F)(F)F)CC1C 85125,Cn1ccn2ncc(C(=O)NCC3CC3CNC(=O)CC3CC4CCC3C4)c12 85126,N1(C(C2CNC(=O)N2)=O)CCC(CNC(c2cnc3n2CCC3)=O)C(F)(F)CC1 85127,C=C(C)C1OCCC1C(=O)NCC1(NC(=O)C(F)C(C)(C)O)CCCC1 85128,N1(C(c2c(CC)scn2)=O)CCC2(CCCN(C(c3nncs3)=O)C2)C1 85129,c1(NC(=O)C=CC(F)(F)F)cncc(CO)c1.C12CCC(C1)NC2=O 85130,c1(C(N(C(CNC(C=CSC)=O)C2CC2)C)=O)cccc(NC(C)C)c1 85131,C1(CCOCCNC(=O)OC(C)(C)C)CCC(=O)NC1.C1CC(=O)N1 85132,CC1CCCC(C(=O)Nc2scc(C(N(C3CN(S(C)(=O)=O)C3)C)=O)n2)C1 85133,C(c1ccncc1)=C(C)C(=O)NCC1CCCCC1NC(C1CCC2CC12)=O 85134,N1(C(CC2N(C(C=CC(=O)OCCCC)=O)CCOC2)=O)CCCC(O)(CC)C1 85135,n1(CC(N2C(CN(C(CC3CC(C)C3)=O)C)CCCC2)=O)nc2c(n1)CCCC2 85136,C1(NC(CC2C(C(=O)OCC)C2)=O)CCCC1NC(c1c[nH]nc1OC)=O 85137,c1(OCC)ccc(-c2cn(CC(C)NC(C3(C4(C)CC4)CC3)=O)nn2)c(F)c1 85138,C1(C(=O)NCC2(CNC(C(C(C)C)C3CCC3)=O)CCC2)Cc2nccn2C1 85139,c1(NC(NCc2c(OC)n(C)nc2C)=S)c[nH]c2ccccc12 85140,c1(CC)nc(Cl)c(CC)c(=NC2CC(NC(=O)C3=C(Cl)CCOC3)C2)[nH]1 85141,N1(C(c2c(C(C)C)ncnc2)=O)CCC(NC(=O)C(O)C(C)(C)C)C12CCCC2 85142,c1(OC)ccc(F)cc1CCC(N1CC(NC(=O)Cc2cncn2C)C(C)C1)=O 85143,C1(C2CC2)(C(N2CC3C(CNC(C4CCS(=O)(=O)N4)=O)C3C2)=O)CC=CC1 85144,C12(CCC(=O)N(CCC(C)NC(C3(CF)CC3)=O)C)CCC(CC1)C2 85145,C1(C(F)F)(CNC(C(C)OCCCC)=O)CCN(C(c2cncc(OC)n2)=O)C1 85146,N1(C(C2CCN(C)S2(=O)=O)=O)CC2(CCN(C(=O)C=CC3CCOC3)CC2)C1 85147,C(=O)(C(C)CC(F)(F)F)NC1CCCCN(C(C2CC(OC)C(OC)C2)=O)C1 85148,CCCC(CNC(C1CC1OC(C)=O)=O)C(=O)NCC(C)(CC)CO 85149,N1(C(C(=C(C)C2CC2)F)=O)CC(CCNC(C2(C)CCN(C)CC2)=O)OC(C)C1 85150,N1(C(C2C3CN(C(CCOCCOC)=O)CC32)=O)CCC(OC)C(O)C1 85151,C1(NC(c2c(C)nn(CC)c2C)=O)CC2CC(C1)CN(C(=O)C(F)C(C)(C)O)C2 85152,C1(C(=O)NCCOC2(C)CCC2)(CNC(CCCSCC=C)=O)CC2(CC2)C1 85153,C(=O)(C(Cl)=CCl)NCC(C1CCOC1)NC(CC1CN(C)C1)=O 85154,C1(NC(c2nc(CC)oc2)=O)CC(CNC(c2ncc(F)cn2)=O)C1(C)C 85155,C=C(C)CC(C)(C)C(=O)N1CC2CCC(C1)C2NC(c1cc2c[nH]nc2s1)=O 85156,Cc1ncc(C#N)c(NC2CN(C(c3ccc(O)c(O)c3Cl)=O)CC2C)n1 85157,C1(NC(c2ccc(C(C)O)cc2)=O)CN(C(c2ccc(C#N)nc2)=O)CC1C#N 85158,C1(NC(C(c2cc(C)sc2)(F)F)=O)CCN(C(=O)C(C)C#N)C(C)C1 85159,Cc1nc(C(N2CCC(C(C)NC(C3(C)SCCCS3)=O)C2)=O)cn1C(F)F 85160,c1(OC)c(C(=O)NC2CC(CNC(=O)CN3CC(C)C3)CC2O)ccnc1F 85161,C(=O)(C1=Cc2ccccc2C1)NC(C(=O)NC(C1CSC1)C)c1ccoc1 85162,C(=O)(C1=NNC(=O)C1)NCC1(NC(CC2C=NN(C)C2=O)=O)CCCCC1 85163,CCC(C(=O)NCC1(NC(=O)C(C)(C)C)CN(C(=O)CCCCOC)C1)N(C)C 85164,Oc1cc(CN=c2[nH]cc(-c3cc[nH]n3)s2)cc(F)c1 85165,N1(C(c2scnc2Cl)=O)CCCN(C(=O)C(O)c2ccco2)CC1 85166,N1(C(C(C2CCC2)OC)=O)CC2CCC1C(CNC(=O)CC1CCCC(C)C1)C2 85167,CC(C(=O)N(CCC(=O)NCCC1CC(=O)N(C)C1)CCCO)C(F)F 85168,N1(C(CC(C(C)OC)NC(C23CCC(CC2F)C3)=O)=O)CCC2(CC1)CSC2 85169,CC1CCn2cc(C(=O)NC3CC4CCC(C3)N4c3nccnc3F)nc2C1 85170,CC1CN(C(=O)C(Cn2cncn2)NC(=O)C(=O)Nc2ncc[nH]2)C(C)C1C 85171,C(C1CCN(C(C2CCCCS2)=O)CC1)=CC(N1CC(CC(=O)OC)C1)=O 85172,Cc1cc(C(N2CCCC(NC(=O)CCS(C)=O)C2)=O)ncc1Cl 85173,N1(C(C(CC)Oc2ccccc2C)=O)CCC2(CCC2NC(=O)CC#N)CC1 85174,Cc1cc(-n2cncn2)ccc1CNC1CNC(=O)C1 85175,CCC(F)(F)CC(=O)N1CCC(C)(C)C1CC(=O)NCCN1CCOCC1 85176,C1(NC(C=C(CCC)C)=O)CC2(CCN(C(c3cncc(OC)n3)=O)C2)C1 85177,C1(CCC)(NC(=O)CCc2cnc(C)s2)CCN(C(=O)CC2CCOC2)CC1 85178,c1(C(=O)OC)cnc(Cl)cc1NCC1CC(C)CN1CCO 85179,c1(CC)noc(C(=O)NCC2(C(N3CCOC(CC(=O)OC(C)C)C3)=O)CC2)c1C 85180,c1(CCC(=O)NC(C(C)NC(COC(C)=O)=O)C)ccc(OC(C)C)cc1 85181,N1(CCc2cn(CC3CCOC3)nn2)CCN(C(C2CSCN2C(C)=O)=O)CC1.CO 85182,c1(C(N2CCC(CNC(C(N(C)C)C3CC3)=O)C2)=O)ccc(CO)cc1F 85183,C1(CN(CCc2c(C)ncs2)Cc2cncnc2)CC(C)CN1Cc1ccccc1 85184,CC1OCCOC1C(N1CCC(CN(c2cnn(N3CCOCC3=O)c2)C)CC1)=O 85185,Cc1cc(C(=O)NC2CCN(C(=O)Cc3nc(Cl)cs3)C2)cc(F)c1 85186,C(=O)(C(CO)N(C)C)NCCC1CN(C(C(C)OC2CCOC2)=O)C1 85187,N12CC3C4CCC(C3C1)N(C4)C(=O)C1CCCN(C1)CC2=O.C1(CNC)CC1Cl 85188,C(=O)(C(C)(F)C(=O)N1CC(CCNC(c2ccc(C(N)=O)[nH]2)=O)(OC)C1)OC 85189,N1(C(C(C2CCCC2)NC(C)=O)=O)CC2CC(N(C)C(C3(F)CCCCC3)=O)C1C2 85190,N1(C(CCCNC(=O)OC)=O)CC(NC(C2(CF)CC2)=O)CC12CCC2 85191,c1(NC(C(=O)NC2CC(N(C)C)C2)CC2CC(F)(F)C2)ccc(N(C)C)cc1 85192,C12(NC(c3cccc[n+]3[O-])=O)CCN(C(=O)C=CCF)CCC1C2 85193,C1(C)(C(=O)NCC(COC)O)CCN(C(c2cccnc2O)=O)C1 85194,C1(C)(CNC(c2c(OC)c[nH]n2)=O)CN(C(=O)COc2ccsc2)C(C)(C)C1 85195,c1(CC)nccnc1C(=O)NC1(C(=O)NCC2CCOC2C)CCCC1 85196,Cc1cncc(C(=O)NC(C)C(C)NC(c2scc(C)c2Br)=O)c1 85197,CC1CCC(C)(CNC2(c3nnnn3Cc3nnn(C)n3)COCCC2C)CC1 85198,Cc1ccc2oc(C(N3CCN(C(=O)OC(C)(C)C)C(CC(F)F)C3)=O)cc2c1 85199,CC1CCN(C(=O)Cc2ccc(Br)cc2)C(CNC(C2CC=CCC2)=O)C1 85200,S(=O)(=O)(CCC(=O)NCCN(C)C(c1ccc(Cl)s1)=O)NCCNC(C)=O 85201,C(CCC(C)C(=O)N(CC(C)NC(=O)Cn1cnccc1=O)C)OC 85202,CC(CNC(=O)CCn1cncn1)CNC(C1CC(N2CCCC2)C1)=O 85203,Nc1cc(F)c(C(=O)NC(CNC(c2cnc(O)s2)=O)C2CCC2)cc1Cl 85204,Cc1c(CC(=O)N(C2CN(C(c3ccoc3C(C)C)=O)C2)C)oc2ccccc12 85205,N1(C(CC(c2ccc(F)cc2)C)=O)C2CCC1(CNC(C1CCC(=O)N1)=O)CC2 85206,CC(C(=O)N=c1cc2ccccn2[nH]1)NC(c1ccc(=N)[nH]n1)=O 85207,C12(NC(CC(=O)OC)=O)COCCC1CN(C(=O)C=C(C)c1ccsc1)C2 85208,N1(C(CCC=C)=O)CCC(C)N(C(=O)CC2CCOC(C)(C)C2)CC1 85209,C1(NC(=O)CC(F)F)CCN(C(=O)CCc2ccc(OC(F)F)cc2)CCC1CO 85210,c1(OC)ncc(C)c(C(=O)NC(C)CNC(c2nc(C3CC3)cs2)=O)c1Cl 85211,c1(NC(=O)NC2CCCN(C(C(CN)O)=O)C2)cc(Cl)ccc1Cl 85212,C#CCC(C)C(=O)N1CCCC1C(C)NC(c1ccc(-c2cscn2)nc1)=O 85213,c1(NC(C(=O)NC(CCCCC)c2ccccc2)=O)cc(F)ccc1NC(C)C 85214,CCC(C)C(C)C(=O)NCc1ccccc1CNC(=O)Cn1cnnc1O 85215,N1(C(=O)CC2CSC2)CCN(C(c2cnccn2)=O)C(CC(F)F)C1 85216,c1(C(=O)NC2COCCN(C(c3c(C)cc(=N)[nH]c3)=O)C2)nc2c(s1)CCCC2 85217,C1(NC(C2N(CCC)CCCC2)=O)CN(C(=O)C=CC(C)C)C2(CCOCC2)C1 85218,c1(C(N)=O)cc(C(=O)NC2(CNC(=O)C(c3ccc(F)cc3)F)CC2)cc(F)c1 85219,CC1CC(NC(C23CC(CF)(CO2)C3)=O)CCN1C(c1cc(Cl)c[nH]1)=O 85220,C(=O)(C(C)(F)C(=O)OC)N(CC(CNC(c1c(CC)ccs1)=O)C)C 85221,C1(C(N2C3C(NC(CNC(CC)=O)=O)CC(C3)C2)=O)CC2(C1)NC(=O)NC2=O 85222,c1(C(=O)OC)sc(C(=O)NCCC2(O)CN(C(C3CC(C)=NO3)=O)C2)cc1C 85223,C(=O)(C1Cc2ccccc21)OCC1CCN(C(c2c(C)nn(C)c2)=O)C(=O)CO1 85224,c1(CC)c(C(=O)NC(C2CCCN2C(C2CC2C2CCC2)=O)(C)C)cnn1CC 85225,C1(C(N(C(CC)CC)CC(C)C)=O)COCCN(C(c2ccc(O)nc2C)=O)C1 85226,CC(C#N)CCC(=O)NCC1CCCN1C(c1cc(-c2cccc(Cl)c2)[nH]n1)=O 85227,N1(CC)CCOC(C(N2CC(O)CC2CNC(=O)C=Cc2cscn2)=O)C1 85228,C1(CC(=O)N(C(C)CC(=O)NC(C)(C)COC(C)C)C)CCCNC1=O 85229,n1(CCC(COC)O)cnc2c(N(CCF)Cc3cccc(Cl)c3Cl)ncnc12 85230,CC1(C)NC(=O)CCC1NC(=O)CC(C(F)(F)F)NC(c1ccncc1N)=O 85231,N1(C(c2ccnc(-n3ccnc3)c2)=O)CCC2CCCC(C2)C1 85232,C1(C)(C(=O)NCC(CCCC)NC(=O)COC)Cc2ccc(C)cc2C(=O)O1 85233,N1(S(CC(C)C)(=O)=O)CC2(CC(CC(=O)NC(c3ccccc3Cl)C)C2)C1 85234,C1(C#N)(C(=O)NCCC(C)NC(c2n[nH]cc2C2CC2)=O)CC2(CCC2)C1 85235,c1(C(=O)NCC2CN(C(Cn3c(=O)ccc(C)n3)=O)C2)nc2ccccn2c1F 85236,CC(C)C(C(=O)NC(C)C(=O)NO)C(C)NC(c1c[nH][nH]c1=N)=O 85237,C(C(C)(CCC)Oc1cccs1)(c1nnnn1CC(F)F)NCCCSCC 85238,c1(C(=O)OCC)ccc(C(=O)NC2(C)CC2)nc1.C1(C(=O)OC)(C(C)C)CC1.C(=O)N 85239,CCCCCC(C)CC(=O)NCC(CC(C)C)NC(c1ncc2[nH]ncc2n1)=O 85240,c1(OC)c(Cl)ccc(C(N2CCC(C3CC3)(NC(=O)CS(C)(=O)=O)C2)=O)c1N 85241,CC1(C(N2CCC(CCCO)CC2)=O)CCCN1C(c1cc(=O)cco1)=O 85242,C(=O)(C(F)(F)C(O)C(C)C)NC(CC)CNC(c1nc2nc(C)ccn2n1)=O 85243,C1(CNC(C(C)=CC)=O)CC2(CO1)CN(C(c1ccc(OC)c(Cl)c1OC)=O)C2 85244,c1(C(=O)Nc2ccc(NC(C(CC)OC)=O)cc2C)cc(C)cc(Br)c1F 85245,c1(C(N(CC(CC)NC(CC(CC)C2CCC2)=O)C)=O)ccc2ncncc2c1 85246,c1(COC)nc2n(n1)CCCC2NC(=O)C(n1cc(CCCOC)nn1)C 85247,C1(C(N2CCC(C)(CNC(c3n(C)ncc3)=O)C2)=O)CCC(S(N)(=O)=O)CC1 85248,CCC(C)(C)C(C)CC(=O)N1CC(C(C)NC(c2c(C)n[nH]c2C)=O)C1 85249,C1(O)(CC)CCC(NC(=O)C(C)C(C)NC(=O)Cc2nonc2C)CC1 85250,C1(NC(CNC(C)=O)=O)CC2CCC(C1C)N2C(C1CCCCS1)=O 85251,C(CC(C)(C)CC(=O)NC(C)(C)C=CC(=O)NC(C1CCCC1O)C)OC 85252,N1(C(C(CC)=CCCC)=O)CC2CC(C)N(C(=O)CC=Cc3ccccc3)C2C1 85253,c1(OC)cccc(C(N2CCN(C(=O)C(O)C(C)(C)C)CC2CC(F)F)=O)c1C 85254,C1(C(=O)NC(C2CCCC2)CNC(c2nc(Cl)cs2)=O)CCNC1=O 85255,C1(NC(c2c(C(C)C)n[nH]c2)=O)CC2CC1N(C(=O)CC(C)F)C2 85256,C(C(C)(C)C(=O)NCC(C)CN(C)C(C1CCCC(=O)C1)=O)NC(C)=O 85257,C(C(N=c1nc(CCOC)[nH]s1)C(C)C)N(C(C(C)(C)NC(=O)NCC=C)=O)C 85258,c1(C(=O)OC)ccc(C(=O)NCC(C)NC(c2nn(C)c(Cl)c2Cl)=O)c(Cl)c1 85259,C1(NC(C(c2c(C)cccc2)C)=O)CC2CC1CN(C(c1ccsc1)=O)C2 85260,c1(C(N2CCC(CCNC(c3cc(CC)sn3)=O)CC2)=O)cn2ccsc2n1 85261,C1(NC(c2ccc(C)n2C)=O)CCCCN(C(C2(C(F)F)CC(=O)C2)=O)C1 85262,C(=O)(C1=CC(O)C(NC(=O)CCc2cncnc2)C1)N(C)C1CC1 85263,C1(=CC(=O)NCC(CNC(c2n(CC)ccn2)=O)(C)O)C2CC3CC(C2)CC1C3 85264,c1(C(N(C(C)CCNC(C2CC2[N+](=O)[O-])=O)C)=O)ccc(Br)nc1O 85265,C1(C(N(CC(C)OC)C)=O)CC2CCN(CCC(=O)Nc3nccs3)CC12 85266,N1(C(C2CC(C)=C(C)CC2)=O)CCC=C(C(=O)N2CCOCC(C)(O)C2)C1 85267,N1(C(CCCSC)=O)CCC2(CCCCC2NC(=O)CCCCCO)C1 85268,CC(C)CC(C(=O)N1CC(S(C)(=O)=O)C1)ONC(C1(C#N)CCCCC1)=O 85269,N1(c2snc(COC)n2)CCCCC(CNC(=O)CCN2CCOCC2)C1 85270,N1(C(C2(CC(C)C)CC2)=O)CCC2C(CCCN2C(c2cnn(CCF)c2)=O)C1 85271,C1(CN(C)C(C2(CNC(=O)CN3CCCC3=O)CC2)=O)CCCCCCC1 85272,C(c1ccc[nH]1)=CC(=O)NC(CNC(CCC)=O)CC 85273,c1(-n2c(-c3c(C)n(C4CCCC4)nc3)nc(CO)n2)ccc(C(F)(F)F)c(Cl)c1 85274,N1(C(C2(C)C(C)(C)C2)=O)CCC(C(N2CCC(CO)(CO)C2)=O)C(O)C1 85275,N1(C(CCC(=O)OC)=O)CCN(C(c2cnnc(O)c2)=O)C2CC12 85276,O=C(C1=CCCS1)NCC(C1CCN(C(C2(F)CCOC2)=O)CC1)F 85277,c1(NC(C)CCOC)ccc(S(=O)(=O)NCC(c2ccco2)O)cc1Br 85278,CC(CC(=O)N1CCC(CN(C(=O)C=Cc2ncc[nH]2)C)C1)P(C)(C)=O 85279,c1(OC)c(C(N2CC3CC2C3NC(c2ocnc2C)=O)=O)cc(Cl)cc1C 85280,N1(C(C2CC(SC)C2)=O)CCn2c(CNC(=O)C(C)=C3CC3)nnc2C1 85281,c1(NC(CC(=O)NC)C)ccc(S(=O)(=O)NCC(C)(C)OC)c(Cl)c1 85282,c1(N2CC(NC(C(C)CC(C)(C)C)=O)CC3(C2)CC3)ncc([N+](=O)[O-])cc1F 85283,C1(CNC(C(Cn2ccc(C)n2)C)=O)CC2(CCOCC2)CN1C(=O)C=C(Cl)Cl 85284,c1(C(C)C)c(N(CCOC(C)(C)C)C(=O)NC2(C)CCS(=O)(=O)C2)cncc1F 85285,C1(CN(C)C(C2(Cl)CC2(F)F)=O)CCN(C(C2(c3cc[nH]n3)CC2)=O)C1 85286,C(=O)(C1CCCc2nc[nH]c21)NCCCN(C(C1CC(C)C1)=O)CCO 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85304,c1(C(N2CC3CN(C(c4c(C)nsc4)=O)CC32)=O)cc2cc[nH]c2cc1Cl 85305,CC(C)(O)C(C)(C)NC(C1CCC(CNC(c2cnn(CCO)c2)=O)CC1)=O 85306,C(CCC(=O)NCCCC1CCCN1C(=O)C(CC)OCC)N(CCC)CC 85307,Cc1cc(C)n(CC(=O)NCc2cc(C(N3CCCC3CCO)=O)on2)n1 85308,c1(N2CC(C)(C)OC(CNC(C3CCCC(F)C3)=O)C2)ncc([N+](=O)[O-])c(=N)[nH]1 85309,c1(CNC(C(C2CN(C(C(n3c(C)ccn3)C)=O)C2)O)=O)ccc(O)nn1 85310,C1(COC)(NC(=O)Cc2nnc(S)n2C)CCN(C(c2c(O)noc2C)=O)CC1 85311,Cn1nnnc1SCCC(=O)NCC1CC(F)(CNC(=O)Cc2cnoc2)C1 85312,C1(C(N2CCC(CC=C)(NC(c3cc(C)sc3C)=O)C2)=O)CN2CCC1CC2 85313,c1(CCC)nc(=NCCC(C)(C)NC(=O)C(C)c2cccs2)s[nH]1 85314,C1(C(=O)NCC(COC)(C)O)CCCN(C(C2CC3CCCC3C2)=O)CC1 85315,C=CCC(C)(CC)C(=O)N1C(C(=O)NC(C(N)=O)C2CCCC2)CCC12CC2 85316,Cc1ccc([N+](=O)[O-])c(C(=O)NC2CC2NC(=O)COc2ccsc2Cl)c1 85317,N1(C(c2cc(CC(C)C)on2)=O)CCC(NC(=O)CC2CCOC2)C(O)C1 85318,Cc1ncc2c(n1)CCC(NS(=O)(=O)c1ccc(O)cc1)C2 85319,CN1CC(C(=O)NCC(N)=O)C1.C12(CC1)CC(=O)NC2 85320,c1(C(=O)NC23C(CN(C(CC4ON=C(C)C4)=O)C2)CC3)csc2c1CCC(C)C2 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85357,c1(C(=O)NCC2(OC)CN(C(=O)CSCCC#N)C2)ccccc1SC(F)(F)F 85358,C(CCC)(C(=O)N1CCC(C(=O)NCCOCCOC)C1)=CC 85359,C1(CNC(C2CC(OCC)C2)=O)CCCCC1C(N1CC(OC2CC2)C1)=O.C=O 85360,CC(C(=O)NC1CN(C(=O)Cc2ccccc2)C1)C(C)NC(=O)OC(C)(C)C 85361,C(=O)(CCCCC(=O)OC)N1CCC(N(C(CC(CCC)O)=O)CC)CC1 85362,c1(C(=O)NC2C(CNC(CC3(C#N)CC3)=O)CCCC2)nnc2n1CCCC2 85363,C(=O)(C(C)(C)C(C)(C)C)NC1CC(C)(CNC(C2(SC)CC2)=O)C1 85364,C1(NC(N(C(CC)C(C)O)C)=O)CCOC(CNC)C1 85365,c1(C(N2CCC(C(C)(C)NC(c3cn(C)nc3O)=O)C2)=O)c[nH]c2cccnc12 85366,c1(NC(CCCC(=O)NCCC(C)N(C)C(N)=O)=O)ccc(S(N)(=O)=O)cc1 85367,c1(-c2nc(CC(=O)NCCC3=NCC(O)CO3)on2)cnc2cccc(Br)n12 85368,CC(=O)CCN=C(NCC1CC2(C1)CC(C)(C)C2)NCC1CCC2CC1C2(C)C 85369,c1(N(C2CCN(C(C3(C)C=CCC3)=O)CC2)C)ncc2ncnc-2[nH]1 85370,c1(C(=O)NCCC2CSCCN2C(C2CC23CC3)=O)nc(O)[nH]c(=O)n1 85371,C(=O)(CCC(=O)NCC1CC(O)CN1C(=O)CCc1cnc(C)s1)NCCC 85372,c1(OCCOC)ccc(-c2ccc(COc3cnc(Cl)c(C)c3)c(F)c2)c(Cl)c1 85373,CC(CC(C)(F)F)C(=O)NCC1CN(C(=O)CC(F)(F)C(F)F)CCO1 85374,c1(OC)ccc(CC(=O)NCCC(C)NC(=O)C(C)(CO)OC)c(OC)c1 85375,CN1CCCC2CN(C(c3ccnc(Cl)c3Cl)C(=O)NC3CC3)CCC12 85376,C1(CNC(C2C(C)(C)C2)=O)CCCCN1C(=O)Cc1cnsc1 85377,N1(C(c2c(OC(F)F)cc(C)s2)=O)CC2CCC(C1)N2C(=O)CCc1cnn[nH]1 85378,CC1=C(C(=O)N2CC(O)(CCNC(C3CC4CCC(C3)C4)=O)C2)SCCO1 85379,C(=O)(C1=CCC2CCC1N2C(c1cccs1)=O)Nc1c(C)n(C2CC2)nc1 85380,C1(C(=O)NCC(CCOC)NC(COCCCC)=O)CC2CCC(C1)O2 85381,c1(C(N2C(C(=O)NC(CCCC=C)C3CC3)CCC2C2CC2)=O)ccc(F)c(C)c1 85382,Cc1cc(C(N2CCNC(C(=O)NCCC3CCCC3)C2)=O)nn1C 85383,N1(C(C2CC(NC(Cc3n(C)cnc3)=O)C2)=O)CCC2(CCCOC2)C1 85384,C1(C2CCN(C(C3CC3C)=O)CC2)(NC(c2cc(C)cc(Br)c2N)=O)CC1 85385,N1(C(CCN(C(c2n(C=C)nnc2)=O)C)=O)CCN(C)C(C)C1C 85386,CC1CC(NC(c2cc(C(F)(F)F)c[nH]2)=O)CN1C(c1snc(O)c1Cl)=O 85387,c1(NC)ccnc(C(=O)N(CCC(=O)NCc2cc(C)on2)C)c1 85388,CCC(CC(F)(F)F)C(=O)NCC(C1CC1)N(C)C(C1CC2C=CC1C2)=O 85389,Cc1ccc2c(c1)CC(C(=O)NC1CCC(NC(=O)Cn3nccc3C)CC1)S2 85390,c1(CC(=O)N(C(C)CN(C)C(=O)C2CC2)C)ccc(NC(=O)NC2CC2)cc1 85391,C(=O)(C(Cc1cn[nH]c1)N(C(=O)C(C)OCC1CC1)C1CC1)N(CCC)CCO 85392,CCC(F)(F)C(=O)N1CCC(N(C(=O)CN2CC=CC2)CCOC)CC1 85393,c1(C(=O)NC2CC(CNC(C(C)OCC=C)=O)C2)ccc2[nH]cc(C#N)c2c1 85394,CCC(C)C(C)(O)CNC(=O)C(C1CCCC1)NC(=O)CCCn1cccc1 85395,c1(N2CCN(C(C)C(N)=O)CC2)nccc(=NCCc2cccc(Cl)c2)[nH]1 85396,c1(C(=O)NC(CNC(c2ccc(C)cn2)=O)(C)CO)nn(C)c2c1CCCC2 85397,c1(C(N2CC3C(NC(=O)Cc4cc[nH]n4)(C3)C2)=O)ccc(O)cc1O 85398,C1(CC(N2CC(C)(NC(C3C(C)OCCO3)=O)C2)=O)COC2(CCC2)CO1 85399,CC1=C(C(=O)NCc2cc(C(=O)NC34CCCC3C4)on2)CCO1 85400,C1(C(=O)NC2C3CN(C(C(CCC)C#N)=O)C2C3)CCc2nnnn2C1 85401,C(c1cccc(F)c1Cl)=CC(=O)NC(C)(CNC(=O)C1=CCOCC1)C1CCC1 85402,C(CC(C)(C)C(=O)N1CCC(C)C(CNC(=O)CC2CSC2)C1)OC 85403,c1(OC)cccc(C(C)CC(=O)NC(C)CCNC(=O)CCc2ccon2)c1 85404,S(=O)(=O)(c1cccc(=NCc2cc(C(N)=O)no2)[nH]1)NCc1c(COC)cccc1 85405,CC1(C)CC(NC(C2(N3CCOCC3)CCC2)=O)CN1C(=O)C(F)C(F)(F)F 85406,C#CCCC(C(=O)NCC(=O)NCCOC)NC(=O)C(C)SC 85407,c1(NC(=O)OC(C)(C)C)cn(CC)cn1.CC(C(=O)N)NC(=O)COC(F)F 85408,C1(CC(=O)NC2CCN(C(c3ccc(CCC=C)cc3)=O)C2)CC(F)(F)C1(F)F 85409,C1(CCC)CN(C(C2(Cl)CC2(C)C)=O)CCN1C(=O)C=CBr 85410,N1(C(C(C)Oc2ccccc2)=O)CC2CCC(CNC(=O)CC3(C)CCC3)(C2)C1 85411,N1(C(c2cc(CC)c(O)cc2)=O)CC2(CCCC2NC(c2ncccc2F)=O)C1 85412,C(=O)(C(C)S(=O)(=O)C1CCOCC1)NC1CCC(NC(C(C)NC(C)=O)=O)CC1 85413,c1(C(C2CCC2)NC(=O)NC(C)CC2CCC2)ccc(F)cc1F 85414,N1(C(c2c(C)oc(C3CC3)c2)=O)CCCC(c2ccccc2)CC1 85415,c1(NC(C2=C(C)OCC2)=O)ccc(C2=CCN(C(C3CCC(C)O3)=O)CC2)cc1 85416,C(=O)(C(CCF)NC(=O)COCC1CCCO1)N(CCCCC)C 85417,N1(C(C23CC(OC)C2C3)=O)CC2CN(C(c3ccnnc3)=O)CC2C1 85418,CC1CCCN(C(c2cccnc2)=O)C1CNC(C12CC3CC1C2C3)=O 85419,CC1OCCOC1C(=O)NCC1CCCN1C(c1ccc(C(N)=O)s1)=O 85420,CCC(O)CN(C(=O)C(F)OC(F)(F)F)CC1CC1 85421,c1(CC)[nH]c(=N)sc1C(N1CC(NC(=O)Cc2ccnc(F)c2)C(C)C1)=O 85422,Cc1cc(C(=O)NC(C2CCCCN2C(=O)CCSc2nnnn2C)C)ccn1 85423,C(CC(C)C(=O)N1CCCC(C(=O)NCCN2CCOC2=O)C1)=CC 85424,Cc1nc(-c2ccccc2)c(CN2CC(F)CC2C(N2CCCCC2)=O)s1 85425,Cc1ccc(C(=O)NC(CNC(=O)C(Cc2ccccc2)C2CC2)CO)c(Cl)c1 85426,C1(C)(CNC(c2ccn(C)n2)=O)CN(C(=O)CCOC2CC2)CCO1 85427,c1(NC(C2CC(OC)CN2C(=O)Cc2ccc(O)cn2)=O)ccc(O)cc1Br 85428,N12CC=C(CCC1=O)CC2.C1(N(S(CC)(=O)=O)CC(=O)O)CCOC12CCCC2 85429,C#CC1(NC(C2(NC(=O)CN(C)C(C)=O)CCCC2)=O)CCCCCC1 85430,c1(C(N(CCCCNC(C2CCCC2O)=O)C)=O)c(Cl)nc2ccccn12 85431,c1(C(C)NC(C(C)SC(F)(F)F)=O)ccc(CNC(C2(C)CCOC2)=O)cc1 85432,c1(OC)cc(OC)cc(Oc2c(OC)ccc(N3CCC3)c2)c1-c1nccn1-c1ccccc1 85433,c1(-n2c(CN3CCCC3=O)nc(CCCCC)n2)ccc2nccnc2c1 85434,N1(C(C(CC)(C)OC)=O)CCCCC2(CCN(C(C3(CCF)CC3)=O)C2)C1 85435,Cn1ncn(NC(=O)C2CCN(C(C3CCCCCCC3)=O)CC2)c1=S 85436,c1(CN2CCC(N(C)C(c3cc(Br)c[nH]3)=O)C2)cn(CC(C)(C)C)nn1 85437,C(=O)(CCCCCF)NCC1C(NC(c2c(CC)ncs2)=O)C1 85438,C1(CNC(C(=C(C)C2CC2)F)=O)CC12CCN(C(=O)CN1CCOCC1)CC2 85439,C(=O)(C1(C)OCCc2ccccc21)N1CC(CC)(NC(=O)C(C(C)(C)C)SC)C1 85440,Cn1nnc2c1CCN(C(=O)C(C1(C)CC1)NC(C1CCCOC1)=O)C2 85441,C1(C)(C(C)C)C(=O)N1.n1(C(CC)C)c2nnc1SC2.c1(CO)ccc(Cl)cc1 85442,n1(CC)ccc(CC(=O)NC2CCN(C(=O)C(C)(C)c3cscc3Cl)C2)n1 85443,CC1CC(N(C(=O)C(C2CC2)N(C)C(c2ccoc2Cl)=O)C)CC(C)C1 85444,N1(C(C(C)S(N)(=O)=O)=O)CCN(C(C2Cc3ccccc3C2)=O)C2CCCC12 85445,Cc1c(C(=O)N(CCCN(C(=O)CC2(C)CCCCC2)C)C)cnn1CCO 85446,C1(NC(c2c(C)nc(CC(C)C)o2)=O)(CNC(=O)C(C)C#N)CC2CCC1CC2 85447,C(=O)(CCCCCCCCC1CC1)N(C)CCNC(c1nc(Cl)cs1)=O 85448,C1(CCNC(CC(C)C2CC2)=O)CSCCN1C(=O)CCCc1cccs1 85449,N1(C(C=CC=CC)=O)CCC(C)C(CNC(c2cc(C3CCOCC3)[nH]n2)=O)C1 85450,c1(SCC(=O)N(C2CCCN(C(CC(C)NC(N)=O)=O)C2)C)ccc(F)c(F)c1 85451,N1(C(C(C#C)(C)C)=O)CCCN(C(C2CCC(=O)N(C(C)C)C2)=O)CC1 85452,c1(C(N2CC(CN(C)C(c3ncc[nH]3)=O)C2)=O)cn(C)c2ccccc12 85453,C(=O)(CN=S(C)(C)=O)NCC(CNC(C(C(C)O)N(C)C)=O)CO 85454,C(=O)(C(CC(C)C)C(C)C)N1CC(C(C(=O)N(CCCCCC=C)C)O)C1 85455,N1(C(C(=O)NCCOC)CCC2CC=CCC2)CC2CC1CN2C1CC1 85456,C12(C(=O)NC3CCN(C(C4CCSCC4)=O)C3)CC(CO)(C1)OC21COC1 85457,N1(C(CCCC#CC)=O)CC2(CNC(C3CCCSC3)=O)CC1CCO2 85458,C1(CNC(C=CC=CC)=O)CN(C(c2nn(C(C)C)nc2Br)=O)C2CC12 85459,Cc1nc(C(=O)NCC2CC2NC(c2ccn(-c3ccncc3)n2)=O)co1 85460,CC1(C)CCCCC1=CC(N1CC2CC1C2CNC(c1ccc(Cl)o1)=O)=O 85461,CC(CC(F)(F)F)C(=O)N1CC(CO)(NC(C2CC(n3ccnc3)C2)=O)C1 85462,c1(CC(=O)NC(CC2CN(C(CCCC(C)C)=O)C2)C)ccc2cnccc2c1 85463,c1(C(C)(C)C)ccc(NC(c2nccn2-c2ccccn2)=O)o1 85464,c1(C(=O)NCCCNC(C2CC(CC)C2)=O)cc([N+](=O)[O-])cnc1N 85465,Cn1nc(Cl)c(C(N2CCC2CNC(c2nc(Cl)cs2)=O)=O)c1Cl 85466,CC1CC(NC(c2cnc[nH]2)=O)CN(C(=O)Cn2nnc(-c3ccco3)n2)C1 85467,CC1(C)CC(NC(C2CC(C)N2C(C2(Cl)CC2)=O)=O)C1 85468,C(c1scnc1C)=CC(N1C(C(CNC(Cc2c(C)nc[nH]2)=O)(C)C)CCC1)=O 85469,C1(CC)C(NC(c2ncncc2N)=O)CCCN1C(=O)CN(C)C(=O)C1CC1 85470,N1(C(C(COC)NC(C)=O)=O)C2CCC1C(NC(c1ncoc1C1CCC1)=O)C2 85471,C(C(C(C)(C)C)NC(=O)Cn1cccc1)NC(C(C1CCOC1)OC)=O 85472,Cc1nc(C(=O)NC(C)CN(C)C(c2ccc3snnc3c2)=O)ccc1[N+](=O)[O-] 85473,N1(C(=O)NCCc2ccccc2OC(F)(F)F)CC2(CO)CCCC1C2 85474,N1(C(C=COCC)=O)CC(NC(=O)CNC(=O)NC)CC2COCCC12 85475,C=CCC(C)C(=O)NCC(C(C)C)NC(c1cc(C(C)=O)c(C)o1)=O 85476,S(=O)(=O)(c1ccc(C(=O)NCC(O)CNC(c2c(OC)ncnc2C)=O)o1)NC 85477,Cc1scc(CCC(O)CN(C)C)c1C.c1(C(=O)N)ccc(O)cc1 85478,c1(OC)cc(OC)cc(CC(=O)NC2CC(C)CN(C(=O)CC3CN(C)C3)C2)c1 85479,C(C(=O)NNc1ncnc2c1CCC2)c1c(C)cc(C2CC2)cc1 85480,CC1(C2CC2)CCN(C(c2c[nH]nc2CCNC(C2(C)C(C)(C)C2(C)C)=O)=O)C1 85481,c1(CC(N2CCC(C(C)(C)NC(C=CC)=O)C2)=O)c(OC)cc(N)cc1OC 85482,CC(C)CC(=O)NCCC(C)N(C(=O)C(n1cc(Br)cn1)C)C 85483,c1(C(N2CCCCC(NC(C(C)CC3CC3)=O)C2)=O)cc(C#N)c(O)nc1N 85484,c1(OC)ccc(NC(=O)CONC(=O)C=Cc2ccco2)cc1 85485,c1(C(=O)NC(C)CCNC(c2cn(C3CCCCC3)nn2)=O)cccn(C)c1=O 85486,C1(CNC(c2c(OC)n[nH]c2)=O)CN(C(c2ccccc2C)=O)C2(CCC2)C1 85487,C1(NC(CCCc2scc(C)n2)=O)CN(C(=O)CC2CC2(Cl)Cl)C2CCCCC12 85488,C1(NC(=O)CCF)COC2(CCN(C(=O)CC3CCCCCC3)C2)C1 85489,c1(N2CC3CC(NC(C(CC)C)=O)CC3C2)ncc(C(=O)OC)cc1[N+](=O)[O-] 85490,CC1CC(C(=O)NCC(C2CCCN2C(=O)Cn2nccn2)(C)C)CCS1(=O)=O 85491,c1(C(N2CCC(C(=O)OCC)(CC)CC2)=O)[nH]c2nccc-2cc1Cl 85492,N(C1CCCc2nc(C)sc21)C(c1c(OC)n(-c2ccccc2)nc1)c1nn[nH]n1 85493,N1(C(C(n2cc(CCC(C)=O)nn2)C)=O)CC2CCC(C1)O2 85494,N1(CCC)CCC(NC(=O)Cc2ccc(Cl)cc2)CC1.C12CCC1C(=O)NC2 85495,c1(NC(C(C)N(C(=O)C(c2ccccc2)C)CC)=O)cccc(OC)c1C 85496,c1(CCN(C(c2cscc2Cl)C(=O)NCC)CCc2cccs2)ccccc1Cl 85497,c1(SC)cc(N2CCCC(C(=O)Nc3ccc(-c4cc[nH]n4)cc3)C2)ncn1 85498,c1(C(=O)NCC(CO)NC(c2c(C)nc(CC)s2)=O)nc(C)n(C)c1C 85499,C1(C(=O)NCC2CC(NC(=O)Cc3cnn(C(F)F)c3)C2)CCc2nncn2C1 85500,C(CCCC(=O)N1CCCCCC1)N(C)C(c1cccn1C)=O 85501,c1(CCC(=O)NC2CC2C(=O)NCc2cc(F)cc(F)c2)ccc2c(c1)OCO2 85502,Cc1cccn2nc(C(=O)NCC(C)N(C(=O)CCC3CC3(Cl)Cl)C)cc12 85503,C(=O)(NN1CCCC1C(=O)N(C1CCCCC1)CC)C1C(CC)N(C)CC1 85504,c1(C(C)(C)OC)nc(=NCC2(c3ccc(C)cc3)CC2)s[nH]1 85505,c1(C(N2CCCC(C3(C)N=N3)C2)=O)cc2cc(C#N)ncc2[nH]1 85506,Cc1cnc(C(=O)NC(CNC(c2cnc(C3CC3)nc2C)=O)CO)c(Br)c1 85507,c1(C(=O)NCC2C(CNC(C3CCC(C)(O)CC3)=O)C2)cc2n(n1)CC(F)C2 85508,C(=O)(CS(=O)C(F)(F)F)N1CC(CNC(C=Cc2c(C)ccs2)=O)C1 85509,c1(-c2c(-c3cn(CCC=C)nn3)cccc2)ccc(F)cc1F 85510,N1(C(C2(C)CCN(C)C2)=O)CC(C2CCCN(C(=O)C(C)(C)CS(N)(=O)=O)C2)C1 85511,Cc1cc(C(=O)NC2(CC(=O)NC3CC(O)C3(C)C)CCCC2)c2n[nH]cc2c1 85512,Cc1n[nH]c(C)c1CC(C)C(=O)NCC(O)CN(C(=O)CSCC(N)=O)C 85513,C1(C(=O)NC(c2cncnc2)C)C2CC(O)C(C2)N1C(c1cc2n(n1)CCO2)=O 85514,C(=O)(C(CC(C)(C)C)OCC)N(CCCNC(C1COCOC1)=O)CCC 85515,c1(OC)cc(OC)cc(C(N2CC(C(C)NC(C3CCCC3(C)C)=O)C2)=O)c1 85516,N1(C(CC(CC)(C)C)=O)CCCC2(CCN(C(=O)Cn3cc(CO)nn3)CC2)C1 85517,C1(C(N2CCC2CC2CC2)=O)C(C2CC2)CCN1C(C1CCCCCC1)=O 85518,Cc1ncc(C(=O)NC2CCCC2NC(C2CCCN2C(=O)C(C)CSC)=O)[nH]1 85519,c1(C(N2C(CNC(c3ccoc3Cl)=O)C=CC2)=O)cc(O)c2ccoc2c1 85520,C1(C(=O)NC)(COC)CCN(C(=O)CC2(CCCN(C(C)C)CC)CC2)C1 85521,c1(C(=O)NC23CCCC2CN(C(c2cc(O)cs2)=O)C3)cnc(O)c2ccsc12 85522,CC(C)(C)CCC(F)C(=O)N1CC(CNC(=O)C=C2CCOCC2)C2(CCC2)C1 85523,C(=O)(C(C)(C)CN(C(=O)CC(C)COC)C)NCc1cc(CC)no1 85524,C(C(O)C(F)(F)F)NC(CC1N(C(C2C(C)(C)C2)=O)CC1)=O 85525,c1(NC(N(CCO)Cc2scc(C)n2)=O)ccc(I)cc1Cl 85526,c1(CC)ccc(NC(=O)CN2CC(c3ccc(F)cc3)C(N)C2)cc1 85527,c1(SC)ncc(N)c(C(=O)NC2CCN(C(=O)C(=O)NCCC(N)=O)C(C)C2)n1 85528,c1(N2CCC(CC)(CC)CC2)nc(NCC2(C)CCCCO2)c2ncsc2n1 85529,C(=O)(C(C(C)(C)C)NC(c1cc(OC)ccc1N)=O)NCC(CC)OC(C)C 85530,CC1(C)CN(C(=O)COC2CCCOC2)CC1C(=O)NCCn1cccnc1=O 85531,c1(C(=O)OCC2OCCC(C)(C)C2)ccn2[nH]c(=N)nc2c1 85532,Cc1c(Br)ccc(NC(=O)CC2CC(NCc3ccc(CO)cc3)C2)c1F 85533,C(CC(=O)N(CC(O)CN(C)C(C12CC(C(C)C)(C1)C2)=O)C)(OCC)OCC 85534,c1(OC)c(F)cc(C(=O)NCC2CC2NC(=O)C(C2CC2)C2CC2)cc1Br 85535,C1(CNC(C=Cc2ccc(C)nc2)=O)CN(C(c2ns[nH]c2=O)=O)CC(C)(C)C1 85536,c1(C(C)NC(c2n(CC)ncn2)=O)ccc(CNC(C2CC2C2CC2)=O)cc1 85537,CC(CC(=O)NCC12CCCC(CN1C(C1CCC1)=O)C2)CC(F)(F)F 85538,CC(C)C(C(=O)NC1CN(C(=O)C=CCO)CC1F)N1CCN(C)CC1 85539,C(CCCCCN=c1[nH]c2ccc(F)cc2o1)NC(C(CC)SC)=O 85540,C=CCC(CNC(c1c[nH]c(C(N)=O)c1)=O)NC(c1occc1C1CC1)=O 85541,c1(NC2CCC3CN(C(CC4C(C)CCC4)=O)CC32)nc2ccc(O)cc2s1 85542,CCC(CC(=O)N1CC(C(=O)NCCC(C)C(C)C)C2(CCC2)C1)C(C)(C)C 85543,N1(C(C(CCC)OCC)=O)CCC(C)(C)CC1C(=O)NCc1cc(C)nc(C)c1 85544,Cc1c(S(=O)(=O)N2CCCC(C)CC2)sc2cc(F)ccc12 85545,c1(C(N(C2CN(C(CC(C)C3CC3)=O)CC2O)C)=O)cc2c(cnn2C)nc1O 85546,N1(C(C23CCC(OC)C2CC3)=O)CCN(C(c2c[nH]cc2Br)=O)C2(CC2)C1 85547,CC1=C(C)CC(C)(NC(c2sccc2CNC(=O)C2CC2)=O)CC1 85548,c1(C(N2CCC(NC(c3n(CC)nnc3)=O)(CO)C2)=O)c(OC)ccnc1O 85549,Cc1cn2cc(C(=O)NCC(CC(C)C)NC(=O)C(C)n3cnnn3)sc2n1 85550,Cc1cc(C)c2nc(N(C3CCN(C(C4(O)CCSC4)=O)C3)C)sc2c1 85551,c1(C(=O)NCC(c2ccccc2)CNC(C(CCC)OC)=O)c(N)sc(C)c1C 85552,Cc1cc(Cl)nc(N)c1C(N1CCCC(O)(CNC(=O)CC2CCCC2O)C1)=O 85553,c1(C(C)=O)ccccc1OCC(=O)NCC(C)(C)CNC(=O)C=CCO 85554,c1(CC(=O)NCC2(C)CCCN2C(c2csc(C3CC3)n2)=O)ncn2c1CCC2 85555,c1(NCc2cc(C)ncn2)nc(N2CC3CC3C2)nc2sccc12 85556,C1(C)(NC(c2ncn(C)c2)=O)CCN(C(c2nnc(C(C)(C)C)s2)=O)C1 85557,N1(C(C2N(C)C(=O)CC2)=O)C2CC=C(C(=O)NCc3n[nH]c4c3CCC4)C1CC2 85558,c1(C(N(C(CN(C(c2nc(C(C)=O)sc2)=O)C)C)C)=O)ccc2sncc2c1 85559,Cn1ncc(Br)c1C(C(=O)NC1(C)CC1)N1CCC1c1cccc(Cl)c1 85560,N1(C(CC(C)C)=O)CCCC(CN(C(=O)Cc2ccccc2F)C)C1 85561,N1(Cc2c(CC)noc2CC)CCC(NC(=O)CC2CCCC2(F)F)C(C)C1 85562,C#Cc1ccc(NC(N2CC(C)(c3ccccc3)C2)=O)cc1Cl 85563,C1(CNC(c2c(C)nc(O)[nH]2)=O)CCC12CCN(C(=O)Cc1csc(Cl)c1)CC2 85564,C1(N(CCCc2nccc(C)c2)CC(=O)OC(C)(C)C)CCC2(CC1)CNC2 85565,Cc1cc(C(=O)NC2CCC(NC(c3ccc(O)nc3C)=O)C2)cnc1C 85566,C=C(C)CN=C(NCc1ccc(Cl)cc1Br)N(C)Cc1ccc(OCC)c(O)c1 85567,C1(C(=O)NC(CC)CN(C(=O)C(C)C)C)CC(c2cnn(C)c2)=NO1 85568,C#CC1(O)CCN(C(C2(CC=C)CCN(C(=O)CC(C)(C)C3CC3)C2)=O)C1 85569,Cc1ccc(O)c(NC(C2(CNC(C3CC3C(=O)N(C)C)=O)CC=CC2)=O)c1 85570,Cc1ccc(C(=O)NC23CCN(C(c4csc(C(F)F)n4)=O)CC2C3)nc1C 85571,N1(C(C2CC(OC)C2)=O)CCCC(C)C1CNC(c1cnn(C)c1Cl)=O 85572,Cn1ccc2[nH]c(C(=O)NCC3CN(C(=O)CC45COC(C)(C4)C5)CCO3)cc12 85573,N1(C(c2c(OC)n[nH]c2)=O)CCC2(CC1)CC2CNC(C1CC(F)C(=O)N1)=O 85574,c1(NC(C2N(Cc3c(F)ccc(C)c3F)CC(O)C2)=O)cccc2c1CNC2=O 85575,NCC(C(F)(F)C(F)(F)F)NC1CCCCC1c1ccccc1 85576,S(=O)(=O)(c1c[nH]ccc1=NCCn1cnc(C)c1C)NC(C=C)(C)CC 85577,c1(OCCNC(N(CC(C)C)CCC)=O)cc(O)ncc1Br 85578,C1(CCNC(C(=O)Nc2cccc(N3CCN(C)C3=O)c2)=O)CCC(F)(F)CC1 85579,C(CC(O)C1CC1)N(CC=C(C)C)CC1(C#N)CC1 85580,c1(C(=O)NCC2(F)CC(CNC(C3C(C)C3)=O)C2)ccc2nc(=N)[nH]n2c1 85581,C=CCCCC(C)(C)C(=O)NC1CCCC(NC(c2ccccc2CC)=O)CC1 85582,C1(NC(Cc2cnc(C)o2)=O)C(C)CCN(C(=O)CCS(N)(=O)=O)C1C 85583,Cc1cn2cc(C(N3CCC(CO)(NC(C4COCCO4)=O)C3)=O)ccc2n1 85584,N1(C(C(C2CCCO2)OC)=O)CCN(CCNC(c2cnc(C)s2)=O)CC1 85585,c1(OCC)ncc(C(=O)NCC2CCCN(C(C3(C)CCCO3)=O)C2)cc1Cl 85586,C=CCCCCCCCCC(=O)NC1CC(F)CN(C(c2cc(Cl)n(C)n2)=O)C1 85587,c1(C(=O)NC2CC(CCNC(COC)=O)C2)cc(C2CC2)nc2onc(C)c12 85588,CC(O)C(F)(F)C(=O)NC1(c2ccc(Br)cc2)CN(C(=O)C(N)=O)C1 85589,Cn1nccc1C(F)=CC(=O)NC12CC1CN(C(=O)CSc1n[nH]c(O)n1)C2 85590,N1(C(C(CC#C)CC#C)=O)CC2(C1)CN(C(=O)COCC1CC1)CCO2 85591,N1(C(C2(NC(C(CC=C)C)=O)CC(O)C2)=O)CC2CN(C)CC2C1 85592,Cc1nc(C2CC2)nc(C)c1C(=O)NCC(F)CNC(C1CC1(Cl)Cl)=O 85593,C1(NC(C2C(NC(C3CCCC(=O)C3)=O)CCCCC2)=O)CCn2ncnc2C1 85594,C(=O)(C(C(F)(F)F)C(F)(F)F)N1CCC2(C(CNC(CC(CC)CC)=O)C2)CC1 85595,C1(CCNC(C2(CC=C)CC=CC2)=O)CCCN(C(=O)CC2C(C)C2(F)F)CC1 85596,C12(NC(C(C)CF)=O)CCCC1N(C(c1ccnc(S)c1)=O)CC2 85597,c1(C(N(C(CNC(C2CN(C(C)=O)C2)=O)C2CC2)C)=O)cc([N+](=O)[O-])cnc1O 85598,C(C(CNC(=O)C(=O)NCC(F)F)S(C)(=O)=O)NC(C1(CO)CC(C)(C)C1)=O 85599,N1(C(c2c(C)con2)=O)CCCC(c2n[nH]c(CNC(=O)Cc3cccs3)n2)C1 85600,C(CC(C)C(=O)N(C1CCCN(C(c2ccccc2NCCO)=O)C1)C)OC 85601,N1(C(C2C(CC)C2)=O)CC(CNC(c2cnnn2CC)=O)(COC)C1 85602,C1(NC(=O)CC2CCCN2C(C2(COC)CCCC2)=O)CC2CC(N)CC12 85603,CCCC(C)(CCC)C(=O)N1CC2CCN(C(c3[nH]nnc3C)=O)C2C1 85604,c1(C(=O)NCC2C(NC(COC(CC)(C)C)=O)C2)ccc(OC)c(F)c1 85605,N1(C(c2c(C)ccs2)=O)CC2(CC2)CC1CNC(C1CC2CC1CO2)=O 85606,c1(C(=O)NCC2CC(NC(c3c[nH]c(=NC)o3)=O)C2)cc(NC(C)=O)cnc1C 85607,N1(C(CC(=O)OCC)=O)CC(F)CC1CN(C)C(c1ccccc1)=O 85608,c1(CN(C)C)ccc(C(=O)NC(c2ccccc2)CNC(C2(Br)CC2)=O)cn1 85609,c1(OC)cc(C)ccc1NC(C12CC(CO1)N(C(c1ccnc(O)c1)=O)C2)=O 85610,N1(C(C(C)(C)OCC)=O)CCC2(NC(=O)CN3OC(C)(C)CC3=O)CC2C1 85611,C(=O)(CC(C)(C)C)C(C#CCNC(C)=O)=O.C(C(C)(C)C(C)O)N 85612,C(Cc1ccccc1)(C(=O)NC(C)(C)CNC(C1CC(CCF)C1)=O)NC(C)=O 85613,N1(C(c2c(C(C)C)ncs2)=O)CC2CC(NC(=O)CCCCCF)CC1C2 85614,C#CCC(C(=O)N(CCCC(F)(F)F)C)NC(C1CCC(OC)CC1)=O 85615,C(C(C(=O)N(C1CCC(C)(C)CC1)C)C(C)C)NC(c1c(C(C)C)c[nH]c1)=O 85616,c1(CNC(c2cn(C)nn2)c2nnnn2CN2CCOCC2)cccc(CO)n1 85617,N1(C(C(CCC)O)=O)CCCC(C)(NC(c2occc2Cl)=O)C1 85618,O=C1CCCCC(C(N2CCC2CNC(C2CC(O)C2)=O)=O)N1 85619,c1(C(=O)NCC(CNC(c2cc(F)n(C)n2)=O)OC)cc(F)c2ncccc2c1 85620,Cc1ccc(=O)n(CC(N2CCC23CN(C(C2CC24CCOC4)=O)C3)=O)n1 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85655,C(=O)(C(CO)C(C)(C)C)NCC1(C(C)NC(=O)CCCn2cc(CO)nn2)CC1 85656,N1(C(C(=O)NC2CC2)=O)CCCCC1C(=O)NCC1(c2cccc(F)c2)CCC1 85657,c1(NC2CC(NC(C3(F)CCCC3)=O)C2)nccc(Oc2ccccc2)n1 85658,CON(CCC(=O)NC)C(=O)C(C)N1CCCC1.C1(CC(C)C)CC(F)(F)C1 85659,C1(C(=O)OCC)CC(NC(=O)Nc2cccc3nc[nH]c23)C2OC(C)(C)OC12 85660,N1(C(C2(OC)CCCCC2)=O)CCCN(C(C2CCCC(C)(C)C2)=O)CC1 85661,c1(C(N2CCN(C(C(C=C)(C)O)=O)CC2CCO)=O)n[nH]c2ccc(C)cc12 85662,N1(C(=O)C=CC2CCCC2)CCN(C(c2ccc(CF)cc2)=O)C(CCO)C1 85663,N1(C(CC(CNC(C(CC)(C)OC)=O)O)=O)CCC2(CCC2)C1 85664,Cc1cc(=NC2COCC2F)[nH]c(=NCc2ccc(CN(S(C)(=O)=O)C)cc2)[nH]1 85665,c1(-c2nc(CCN(C)C)nn2CC2CCCO2)ccc2ncc(I)n2c1 85666,C1(CCNC(c2onc(CC)n2)=O)CCCCN1C(c1conc1COC)=O 85667,CCC(C)C(O)C(=O)NC1(COC)CCN(C(c2cn(C)nc2Br)=O)CC1 85668,c12ccc(C)c(c1)C(=O)NCc1cn-2nn1.Cc1cc(C)n(CC(C)N(C)C)n1 85669,C12CCN(C(=O)CNC1=O)O2.C1(C(C)C)CCN1C(N)=O 85670,C(c1cnc(O)nc1O)=CC(=O)N(CCN(C(=O)CC1(CS(C)(=O)=O)CC1)C)C 85671,CCC(Cc1ccc(N)cc1)C(=O)NCCNC(=O)CCc1nnc(C(F)F)o1 85672,c1(-c2c(COC)n[nH]c2)nc(C2CCCO2)nn1CC1CCSC1 85673,c1(C(=O)NCC2(F)CC(NC(CN(C)C)=O)C2)cccc(-n2ccnc2O)c1 85674,C1(NC(=O)CC2OCCO2)CC2(CCOC2)C1 85675,c1(NC(N2CC(C3CC3)C2)=O)ccc2nc(CO)[nH]c2c1 85676,C1(C(=O)NC(c2ccc(F)cc2)CNC(C(CO)N(C)C)=O)CSCC(=O)N1 85677,c1(C(N2CC3(CC(C(=O)Nc4ccon4)C3)C2)=O)ccc(Cl)cc1OCF 85678,CC1=NOC(C)(C(N2CC(C)(NC(c3cc(C)c(-c4ccccc4)s3)=O)C2)=O)C1 85679,c1(NC(C2(C)N(Cc3n(C)cc(Br)n3)CC2)=O)cnc2cccnc2c1Cl 85680,C1(CC)CN(C(c2cnc(C3CC3)[nH]2)=O)CCN1C(c1cccc(C(F)F)c1)=O 85681,C1(NC(COC2CCN(C(c3n(C)nnc3)=O)C2)=O)CCCCCCC1 85682,C(CCN(C)C(C1(C)CC=CC1)=O)(C(C)(C)C)NC(C(c1ccccc1Cl)C)=O 85683,C1(NC(c2ccc(OC)cc2F)=O)CCCCN(C(=O)C(=O)NC2CC2)CC1 85684,C1(C(=O)NCCCN(C(=O)CCc2cccn2C)CC)CCNC1=O 85685,C1(C(N2C(c3cn(CC(=O)OCC)nn3)C(C)CC2)=O)CCn2cnnc2C1 85686,c1(NC(=O)NC2(C3CCC3)CCC2)ncc(C(F)F)cc1Cl 85687,N1(C(C(C(C)C)SC)=O)CCC2(CC1)CCN(C(C1CCC3CCCCN13)=O)C2 85688,Cc1nc(N2CCC(C3CC3)C2CNC(C2(CF)CCC2)=O)c2scc(C)c2n1 85689,C1(NC(C2(CCNC(=O)CC34CCCC3C4)CCCC2)=O)CC2CC1C(O)C2O 85690,c1(N(C(CNC(C(C)=CC)=O)C)CC)nc2ccc(C(=O)OC)cc2o1 85691,N1(C(C(CCC)C)=O)CCCC(CNCc2ccc(Cl)cc2C(C)C(=O)O)CC1 85692,C(=O)(C(C)(O)C(C)C)N(C)CC1N(C(c2cc(CCOC)on2)=O)CCCC1 85693,C1(=CC(=O)NC(C2CCCC2)CNC(C(CCSC)O)=O)CCCCC1(C)C 85694,c1(CNC(CN(S(CC)(=O)=O)C2CC2)=O)ccc2c(c1)oc(=O)n2C 85695,Cc1cc(C(N2CCN(C(=O)C(F)n3cccn3)C(C)C2)=O)cc(C)c1 85696,c1(CC(=O)NC(C2CC=CCC2)C(=O)N(CCCOC)CCO)ccnc(O)c1 85697,c1(C(N(C2CCN(C(CC3CC(CC)C3)=O)C2)CC)=O)c(C)noc1Cl 85698,C1(NC(C2N(C(C)C)CCC2)=O)COC2(C1)CN(C(c1cncs1)=O)C2 85699,C(=O)(C1CCOc2ccc(Br)cc21)N1C(c2cn(C)nc2)C(=O)NCC1 85700,C1(C)(CC)CC(Oc2ccc(C(=O)OC)cn2)CN1C(=O)C(C)C 85701,N1(C(c2c(CCCC)ocn2)=O)CC(NC(c2cnc(O)c(Cl)c2)=O)CC(O)C1 85702,C12CN(CCO1)C2=O.C1(CN(C)C)CCC(NCc2cccnc2)CO1 85703,C(=O)(CC(C)CC(C)C)NC1CC(NC(CNC(=O)NC)=O)CC1O 85704,CC(C)C(C(C1CCCCC1)NC(=O)CC1CCCC1)NC(c1nc(Cl)cs1)=O 85705,C1(CNC(CC=C=C)=O)CCN(C(c2cc(Cl)cc(F)c2F)=O)CCC1(F)F 85706,C1(N(c2n[nH]c3c2CCC3)C(c2ccccn2)=O)CCC2(CCNC2)CC1 85707,C1(C#N)(COC)CN(C(=O)C(C2(C)CC2)NC(=O)Cc2cccnc2O)C1 85708,N(C1CCc2c(Cl)ccc(Br)c21)S(c1c(C)cccc1Cl)(=O)=O 85709,C(=O)(CCC(C)N(C)C)NCCN(C(=O)C(F)(F)c1csc(Cl)c1)CCC 85710,C12(C(=O)NC3(C)CN(C(c4ccn(C)c(=O)c4)=O)C3)CC(C)(C1)OC21COC1 85711,C1(CNC(CN(C(COC)=O)C)=O)C(C)CCCN1C(c1scnc1Cl)=O 85712,c1(C(=O)NCCCCCNC(=O)C=Cc2ccccc2)c[nH]c2c(F)cccc12 85713,C1(C(=O)NCC(CC)(CC)NC(c2cnccc2OC)=O)CC2(CCCC2)CO1 85714,c1(C(c2n(C(CC)C)nnn2)NCc2cnc(Cl)s2)ccc(C2CC2)cc1 85715,Cc1ncc(CNC(C2CCN(C(C3(O)CCOC3)=O)C2)=O)o1 85716,CCC(CCC(=O)N1CCCC(C(N2CCN(C)CC2CO)=O)C1)OC 85717,C1(C(C)CNC(C2CC=CCC2)=O)CCN(C(CC(C)(C)C)=O)CC1 85718,CC1CC(NC(=NCCNC(=O)OC(C)(C)C)NCCC(F)(F)F)CCN1C 85719,c1(C(=O)NCCCN(C)C(C2CCCN2C2CCOCC2)=O)ccncc1N 85720,c1(NC(C(C)(C)NC(c2cn(CC)nc2)=O)=O)cn(C)nc1C 85721,Cc1nocc1CNC(C1(NC(=O)CCc2ccccc2)CC1C)=O 85722,c1(C(C)C)[nH]ccc1C(N1CCC(C(=O)NCC(O)CC2CCC2)C1)=O 85723,C(C)(CCCC(C)C)NC(CC1(COC)CCOC1)=O 85724,CN=c1ccc(C(=O)NC2(C(N3CCC3C(N)=O)=O)CCCC2C)c[nH]1 85725,C1(OC)CN(C(=O)Cc2n[nH]c(C)n2)CC1NC(=O)CCOC1CCCC1 85726,c1(CCNC(C(c2ccco2)NC(COC(CC)C)=O)=O)c[nH]nc1O 85727,c1(-n2c(C3CCC(OC)C3)nc(-c3ccoc3C)n2)cc(F)cc(F)c1 85728,C1(C(N2CC3C(CCNC(=O)C4=CCCCO4)(CC3)C2)=O)CCC2(CCC2)CC1 85729,C=CC(C)(CC)C(=O)NC1C2CC1N(C(c1ccsc1OC)=O)C2 85730,C(=O)(C1(C)CCn2ccnc21)N1CCC(O)(CN(C)C(C2CCCC(F)C2)=O)C1 85731,Cc1cc(=NC2C(C)C2C)[nH]c(N2CCOC(c3ccc(C)s3)C2)n1 85732,c1(OC)cc(C(N2CC(NC(=O)Cn3cccn3)C(F)C2)=O)cc([N+](=O)[O-])c1C 85733,C1(C)(CNC(CC(=O)OCC)=O)CCN(C(=O)C(C(C)O)N(C)C)C1 85734,c1(C(=O)NC2(CO)CN(C(C(CN(CC)CC)F)=O)C2)cccc(COC)c1 85735,C(=O)(CC(=O)N1CC(NC(C2CC(OC)C2)=O)C1)OCC 85736,c1(C(=O)OC)cc(C(N2CCC(CNC(=O)COc3ccsn3)C2)=O)cc(F)c1 85737,C1(NC(CCC#CC)=O)CN(C(c2cccc3ccoc23)=O)C2(CCCC2)C1 85738,CCCC(C)CC(=O)N1CCCC1CN(C(=O)C(C1CCOCC1)=O)C 85739,c1(C(=O)NC(C)(C)CNC(=O)C=CC(=O)NC2CC2)ccc(C(O)CF)cc1 85740,n1(CC(=O)NCC(c2ccc(OC)c(OC)c2)C)sc2cccnc2c1=O 85741,Cc1cc(C(=O)NCC2CC2CNC(c2ccccc2F)=O)cc(C)n1 85742,C(C#Cc1cccnc1)Oc1ccccc1.c12cccc(c1)CNC2=O 85743,Cc1ncc(CCC(N2CCN(C(=O)CCNS(C)(=O)=O)C3CC23)=O)c(O)n1 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85849,c1(OC)ccc(C)cc1C=CC(N1CCCCC1CNC(c1n[nH]cc1C)=O)=O 85850,N1(C(C2CC3CC3N2C(=O)CCN2CCCCC2)=O)CC2(CCOC2=O)C1 85851,c1(C(=O)OC)coc2c1CN(C(=O)C=CC1CCC1)C2 85852,C1(NC(C2C(=C)C2C(=O)OC)=O)CN(C(=O)C2=CSCS2)CC1C(F)F 85853,N1(CC(=O)NC(C(=O)N(CC(CCC)O)C)CC2CCC2)CCC(=O)CC1 85854,C1(C(=O)NC(CNC(C(Cc2ccc(OC)cc2)O)=O)(C)C)CCN(C)S1(=O)=O 85855,C1(C(=O)NCCC(C)CCNC(=O)COC2(C)CCC2)(OC)CCC12CCC2 85856,N1(C(c2cc(CCC)oc2C)=O)CCC(C)C(N(C(=O)C(C)OCC(C)C)C)C1 85857,c1(NC(C2N(C(CCOCC#C)=O)CCCC2)=O)ccc2oc(C(N)=O)cc2c1 85858,c1(NCC(C(CC)CC)OC)nccc(=NCCN2CCCC2)[nH]1 85859,C12(C(=O)NC3CN(C(C4C(Cl)(C(=O)OCC)C4)=O)C3)CC(CN1C1CC1)C2 85860,O(N(C)C(=O)CCc1cnc(C)[nH]1)CC(=O)OC 85861,Cc1ccsc1CC(=O)NC1(CNC(=O)C(C)CN(C)C)CCOC1 85862,C1(N(C(CC(C)c2ccco2)=O)CCNC(c2ccn(C)n2)=O)CCCCCC1 85863,C1(c2scc(C)n2)CN(C(=O)Cn2cc(CN(C)C)nn2)CCO1 85864,N1(C(CC(C)=C(C)C)=O)CC(CNC(=O)C(C)Cc2ccccc2)CCC1C 85865,CC1(O)CCN(C(=O)CCCNC(=O)CC2(N(C)C)CCC2)CC1O 85866,N1(C(C(c2nc(F)ccc2Cl)C)=O)CCSCc2ccccc21 85867,C(C)(C)(CCCNC(C1NC(=O)CC1C)=O)NC(COCc1nnc(C)s1)=O 85868,C1(C)(C(=O)NCC(CCC)O)CCN(C(=O)CC(C)C)C1 85869,CCCCC(F)(F)C(=O)NC(CC1CCOCC1)C(=O)NOCC(=O)OCC 85870,C1(S(C)(=O)=O)(C(=O)NC2C(NC(Cn3nc(C)n(CC)c3=O)=O)C2)CCOCC1 85871,c1(OC)c(C)cc(C(=O)NC2CCC(CNC(c3cccc(C)n3)=O)C2)cc1C 85872,C(=O)(NNC(=O)OC1CCOCC1)NCC(C)C.C12CCCCC1O2 85873,C1(N(C(c2c(CNC(Cc3cc(C)[nH]n3)=O)noc2)=O)C)CCCC1(C)O 85874,c1(OC)ccc(C=CC(=O)NC2CCCC2NC(c2cccn2C)=O)c(C)c1 85875,C(=O)(C(CCC1CC1)NC(=O)C(C#N)C1CC1)OC.N1(CC)CC1 85876,C1(C(=O)NC(C2CCCC2)CNC(c2cccnc2F)=O)CC2C=CC1CC2 85877,O(P(C)(=O)CNC(=O)C(Cn1cncn1)NC(=O)C(Cl)Cl)CC 85878,c1(C(=O)NC2C(NC(C3CCC(CC)O3)=O)COC2)c(C)[nH]c(C)c1C 85879,O=C(C(O)CC(F)F)N1CCN(C(=O)CCC2CCCCO2)CC1 85880,C1(OC)(CNC(=O)CCSc2ccccn2)CN(C(C2CC2(C)C(F)F)=O)C1 85881,N1(C(C(C)=NOCC#N)=O)CCOCC(NC(=O)C(C)SC(C)C)C1 85882,C1(NC(C2CN(C(C)C)C2)=O)CN(C(C2CC3(CSC3)C2)=O)CC1N=[N+]=[N-] 85883,Cc1nc(C)c(C(=O)NC2CN(C(=O)C(C)(C)c3ccc(Cl)s3)CC2C)s1 85884,N1(C(c2n(CCC)ncc2)=O)CC(C(=O)NC2(C)CC3(CC3)C2)CC12CCC2 85885,CCC(C)C(CC(=O)N1CC(C)(CF)C1)NC(C1CC2(CCO1)CC2)=O 85886,C(=O)(C(C)(CS(C)(=O)=O)NC(c1cc(C)sc1C)=O)OC 85887,c1(CC)cccc(CN(C(=O)Nc2nc(C)c(I)s2)C2CC2)c1C(F)(F)F 85888,Cc1cnc(C(=O)NCC2CN(C(c3ccc(CO)cc3F)=O)C2)cc1C 85889,CC(C)CC(C(=O)N(C1CCN(C)C1)C)ONC(=O)C1(C(N)=O)CC1 85890,c1(C(=O)NC2CC(NC(C3(CCCC)CC3)=O)C2)cc[nH]c(=NC)c1[N+](=O)[O-] 85891,C1(OC)CC(CNC(C2CCCC3CC23)=O)N(C(c2ccoc2Cl)=O)C1 85892,C(=O)(CCCC(C)C)NC(CCCC)CNC(c1cn(C)nc1CC(=O)OC)=O 85893,C1(CC(=O)NCc2ccccc2CNC(c2ccncc2)=O)CCC1C1CC1 85894,Cc1c(NCC(C)(C)NC(=O)C(C2(O)CCCC2)F)cccc1C(=O)NS(C)(=O)=O 85895,CC(CCC(C)(C)C)C(=O)N1CC2COCCC2(NC(=O)CCc2cc[nH]n2)C1 85896,N1(C(=O)Cc2cc(Cl)cs2)CCC2(C1)CN(C(c1cncn1C1CC1)=O)CCO2 85897,C(=O)(C1COc2ccccc21)N(CCCN(C)C(c1n[nH]cc1Br)=O)C 85898,C(CC(C(=O)NCCCCC1CC1C)N(C)C)NC(CC1C(CC)C1)=O 85899,N1(C(c2csc(Cl)c2)=O)CCCC(C2CC2NC(C2(CO)CCCO2)=O)C1 85900,c1(C(N2CCC(CN(C(C3CC(OC)C3)=O)C)C2)=O)nc2c(cc1Cl)OCCO2 85901,N1(C(=O)OCC)CCCC1C(=O)NC1CC(NC(=O)CCC=CC(C)C)C1 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86077,c1(C(=O)NCC2(F)CN(C(Cc3scc(C)c3)=O)C2)cnn(C(C)C)c1F 86078,Cc1ccc(CC(N2CCOC(CNC(C3(C#N)CCCC3)=O)C2)=O)c(Cl)c1 86079,C(=O)(C1=CC2C=CC(C1)C2)NC(CC)(CNC(c1[nH]ccc1C)=O)CC 86080,C(CC(O)CC(=O)NCCC1CCCN(C(C)=O)C1)SC 86081,n1(CC)nncc1C(=O)NCCC1(OC)CN(C(=O)C(C)COC)C1 86082,c1(OC)cnc(C(=O)NC2C3CC(NC(C4CC(CC5CC5)C4)=O)CC23)cn1 86083,c1(NC(C23C(CN(c4nc(OC)cc(OC)n4)C2)C3)=O)cc2c[nH]nc2cc1F 86084,C(c1ccccc1)=C(C)C(N1CC(F)CC1C(=O)NCC(c1ccsc1)O)=O 86085,Cc1cc(C(N2CCC=CC2C(=O)NCCCCS(C)=O)=O)cc(C)c1 86086,C(=O)(NNc1cc(F)c(F)cc1Cl)c1cc(OC)c2c(c1)scc2 86087,c1(OCC#C)ccc(C(=O)NCC2CN(C(=O)C(c3ccc(F)cc3)F)C2)cc1 86088,N1(C(C2(C#N)CCOCC2)=O)CCN(C(=O)CC2CCCC(F)(F)C2)C2(CC2)C1 86089,c1(OC)cc(C(=O)N(C2CN(C(=O)CCSc3n[nH]c(C)n3)CC2F)C)nn1C 86090,CC1=C(C(=O)NC2CCN(C(c3ccnc(O)c3F)=O)CCC2CO)SCCO1 86091,c1(CC)ccc(CN(C2C3CN(C(=O)CC(F)(F)F)CC23)CCO)cc1 86092,CC1CCC(C(=O)NC2CC=CCC2)N(C(C2C3CCCC23)=O)C1 86093,c1(OCC(=O)NCCCn2cc(C(c3ccccc3)C)nn2)ccc(I)nc1 86094,Cc1ccc2c(C(=O)N(C)CCn3cc(C4COC(C)(C)O4)nn3)ccnc2c1 86095,c1(CO)nc(Cl)sc1C.C1(CCOC)(C(=O)N2CC2)CC1 86096,C#Cc1cccc(C(=O)NC2(CNC(c3c[nH]nc3C3CC3)=O)CC2)c1 86097,C1(C)(OC(C2CC2)N(C(C2(CC3CC3)CC2)=O)CC)CCCC1(C)C 86098,Cc1sccc1C(=O)NCc1cc(C(=O)NCC(C)C(C)O)n[nH]1 86099,C1(NC(C2(CC)CCC2)=O)CN(C(c2snnc2C2CC2)=O)CCC1C(F)(F)F 86100,c1(C(N(C2CCN(CC3CCc4ncnn43)C2)CC)=O)cc[nH]c2nccc1-2 86101,Cc1c(C(=O)NC2CC(CNC(=O)CCCF)C(O)C2)cc(F)cc1Br 86102,c1(CNC(C(C#C)(C)C)=O)ccc2c(c1)CCN(C(=O)C(C#N)C(C)C)C2 86103,C#CCC(CC(=O)Nc1cnc(OC)nc1)NC(=O)CCC(C)(C)OC 86104,C(=O)(C(C)C(O)C(C)C)N1CCC(C(=O)NCc2snc(C)n2)C1 86105,c1(C(=O)NCC2CN(C(C3(Br)CC3)=O)CCO2)nc2ccccn2n1 86106,Cc1ccc(C(=O)NCC=C2CCN(C(=O)Cn3nnc(=N)[nH]3)CC2)cc1CO 86107,N1(CC)CCCC(NC(C2CCCN2C(=O)C(C)NC(N)=O)=O)C1 86108,CCCCC(O)C(C)C(=O)NC1CCN(C(C2C3C4CCC(C4)C23)=O)C1C(C)C 86109,c1(OC)cc(CN2CC(F)(C(=O)Nc3cccc(Br)c3O)C2)c([N+](=O)[O-])cc1O 86110,N1(c2snc(C(C)C)n2)CC(C)(C)CC1CNC(=O)CC(C)c1ccccc1 86111,c1(C(=O)NC(CNC(C2CC(OC)C2)=O)(C)CO)ccc(=O)n(C2CC2)c1 86112,c1(C(=O)NCC(CNC(c2cn(CC)nn2)=O)CO)c[nH]c2c(C)cccc12 86113,Cc1cc(S(=O)(=O)Oc2cc(C(C)(F)F)ccn2)cc([N+](=O)[O-])c1F 86114,N1(C(COCC=C)=O)CC(C2CC2C(=O)NCC2CC2Cl)C1 86115,N1(C(CCCCC=CC)=O)CCC(C2CCN(C(=O)COCCCC)C2)C1 86116,c1(SCC=C)n[nH]c(=NC(=O)N2CCOC(Cc3ccccc3)C2)s1 86117,c1(N(C)CCO)cc(C(N2CCC2CNC(=O)Cc2nnc(S)n2C)=O)ccn1 86118,C(=O)(C1=CCOCC1)N1CCC(CCNC(c2cccc(F)c2F)=O)C1 86119,C1(NC(C(C2CC2)OCC)=O)CC2CN(C(c3sccc3OC(F)F)=O)CC12 86120,N1(C(CCCN(C(C(C)C(C)O)=O)C)=O)CC2CC(C(=O)OC(C)(C)C)CC2C1 86121,c1(CN(CCNC(Cc2ccc(C)o2)=O)C(C2COCCO2)=O)ccc(Cl)nc1 86122,c1(C(=O)NCC(C(C)C)(C)NC(=O)C(C)C2CC2)c(F)cccc1Br 86123,CC#CCC(C(=O)NCC(O)CC1CCCC1)NC(=O)CCc1ncnn1C 86124,C(C1CSc2ccccc21)NC(=NCCOC)NCc1nnc(CCO)s1 86125,C(CCCCCC(=O)NC(C(F)(F)F)C1CC1)n1cc(COCC(C)O)nn1 86126,CCC(CC(=O)NC(C)C(C)C(=O)NCCc1cc(C)on1)C(F)F 86127,C1(C(N2CCC(COCC)C2)=O)C=CCN(C(=O)CCNC(=O)OC)C1 86128,CCCC(C(=O)NC(C1(C)CCN(C(c2ccnc(OCCO)c2)=O)C1)C)OC 86129,Cc1ccc(C(C)C)c(C(N2CC3CC2CC3NC(=O)C#CC(C)C)=O)c1 86130,C1(NC(=O)NNC(=O)C2CC2)CCCC(c2ccccc2)CC1 86131,c1(C(N2C3C(NC(c4ncncc4Cl)=O)CC(C3)C2)=O)cnc2cc[nH]c2c1 86132,C1(NC(C2(COC)CN(C(c3nnccc3C)=O)C2)=O)CN2CCC1(F)CC2 86133,N1(C(CC=C)=O)CCN(C(=O)CCCCc2ccccc2)C2(CC2)C1 86134,C1(C(N(C(C)C(=O)NCC=CCSC)CCC)=O)COCCN1C(=O)OC(C)(C)C 86135,CC1CN(C(C2COCC(=O)N2C)=O)c2ccc(C(F)(F)F)cc2O1 86136,C(=O)(C#CC1CCCCC1)N1CC(CCNC(c2nc(C)sc2)=O)OC(C)C1 86137,CC1CC(CNC(C2(C)C=CCCC2)=O)CCN1C(c1cc2scnc2[nH]1)=O 86138,C(=O)(CCC(C)C)N1C2CCCN1C2.C1(C=O)C2CCC1(c1ccnn1C)C2.CO 86139,C(=O)(CC(O)CC(C)(C)C)N1CCCC(C(=O)NC2(C3CCCC3)CC2)(CC)C1 86140,c1(CC(C(=O)N(CC(CNC(COC(C)=O)=O)O)C)C)c(C)noc1C 86141,CCN=c1[nH]c(C(N2CCN(C(=O)C=Cc3ccncn3)C(C3CC3)C2)=O)cs1 86142,Cc1cc2ccc(C(N3CCCC3C(C)NC(C3CC34CCCC4)=O)=O)cn2c1 86143,CC(C)(C)CCCCCC(=O)N1CCN(C(=O)C#CC2CCC2)CC1C(F)F 86144,O=C(C(O)C(F)(F)c1ccccc1)N1CCC1C1CCCCC1.c12nnc(o1)C2 86145,C(c1cncnc1O)=CC(N1CCN(C(C2(C)C(C)OCC2)=O)CC1)=O 86146,O=C(C(CO)C(F)(F)F)NC(Cn1cncn1)C(=O)NCC1(C2(O)CCC2)CC1 86147,Cc1cc(Cl)cc2cc(C(N3CCC(C)C3CNC(C3(CO)CC3)=O)=O)[nH]c12 86148,C1(CCOC)(NC(CCCOCC)=O)CCN(C(C2CCC(O)CC2)=O)C1 86149,c1(OCC=C)cccnc1C(=O)NCCC1CCC(NC(c2cc(C)c[nH]2)=O)C1 86150,C(CN=c1[nH]c2ccc(S(=O)(=O)NC(C)CC#N)cc2s1)c1nccc(OC)n1 86151,c1(C(=O)NCc2cccc(NC(C3(CC)CCOC3)=O)c2)cc2sccc2[nH]1 86152,Cc1nc(NCC2CCCCN(C(c3cc(CF)on3)=O)C2)ccc1[N+](=O)[O-] 86153,C=C(C)CC(C(=O)OC)NC(C1CC=CC(n2cc(C(CC)OC)nn2)C1)=O 86154,C1(CC)CN(C(=O)C=C(C)C)CCC1NC(C1CC(F)(F)C1(C)C)=O 86155,CC1CC(=O)NCC1C(N1CCCN(C(C23CCC(CC2)CC3)=O)CC1)=O 86156,N1(C(C(=O)NCSc2cccc(F)c2)C2C(C)C2)CCC(C(N)=O)CC1 86157,C1(NC(=O)Cc2ccc(Cl)nc2)CN(C(C2(F)CCC2)=O)CC2(CC2)C1 86158,CC1CN(C(=O)CC2(N(C(=O)C(n3cc(Cl)cn3)C)C)CC2)CC1N(C)C 86159,C1(NC(CC(C)OC)=O)C2CC1N(C(=O)CCc1cncn1C)C2C 86160,C1(OC)CC(CNC(=O)CCCc2ccc(Cl)cc2)N(C(C2CC(C#N)C2)=O)C1 86161,C1(NC(CC(CC=C)NC(c2cncc(C)c2)=O)=O)COC2(CCCC2)C1 86162,N1(c2cccc(S(=O)(=O)N(C)CC3(OC)CCOC3)n2)CCCC2(CCN(C)C2)C1 86163,C1(N(C)C(c2n[nH]cc2Cl)=O)CCCN(C(C2CC23CC3)=O)CC1 86164,C1(N(C)CCNC=O)CC(C(=O)NCCC2(CC)CC2)C1.c1ccsc1 86165,C1(NC(c2ccc(COC)[nH]2)=O)CC2CC(C1)N(C(=O)CC1NC(=O)NC1=O)C2 86166,c1(NS(C)(=O)=O)ccccc1NC(=O)C(N1CCCCC1CO)=O 86167,c1(CC(C)N(CCC(=O)NCC)CCCOCC)ccccc1 86168,N1(C(CC2(CSC)CC2)=O)CCCN(C(=O)Cc2ccnn2C)CC1C 86169,N1(C(CCCC2(NC(=O)C=C(C3CC3)C3CC3)CCC2)=O)CCOCC(C2CC2)C1 86170,c1(C(C)(C)C)noc(CCC(=O)NCC2(NC(c3cc(C(F)F)no3)=O)CC2)n1 86171,C12(C(=O)NC3C(CC=C)CCC3)CC(CN(C(=O)CCNC(=O)OCC)C1)C2 86172,N1(C(c2c(C)cc(=O)n(C)n2)=O)CCC2CN(C(c3cnc[nH]3)=O)CC2C1 86173,C(=O)(CCCNC(=O)CSC1CC1)NC(C1CCC1)C 86174,c1(C(=O)NCCNC(c2c(C)nccc2Cl)=O)ccc([N+](=O)[O-])c(S(N)(=O)=O)c1 86175,N(C(=NC(C)C)NCC(O)Cc1ccc(F)cc1)C1C(C)CC1 86176,Cc1ccc(Cl)c(C(=O)NC(CNC(C2(C(F)F)CC2)=O)CC(C)C)c1N 86177,c1(NC(N2CCC(C=C)(C(=O)O)CC2)=O)ccc2c(c1)ncn2C 86178,C(C)(N=c1[nH]c2c(c(=NCCNC(=O)C3CC3)[nH]1)COC2)c1cc(C)on1 86179,C1(NC(C2(C(=O)OCC)CCO2)=O)CC2CCC(C1)N2C(=O)C(C)CC(F)(F)F 86180,N1(C(C=CCCC)=O)CCCC(CC(=O)Nc2cnn(CCC)c2)CC1 86181,C1(CNc2c(C(=O)OC)ccnc2)(NC(=O)OC(C)(C)C)OC2CCC1CC2 86182,CC1CN(C(=O)CC2CSC2)CCC1CNC(=O)C=CCOc1ncccn1 86183,C1(C(=O)NCC(C)N(C(c2[nH]cc(C)c2)=O)C)CCCCN1C(C1CCCC1)=O 86184,c1(C(N(C(C)CC(=O)NOCC(=O)N(C)C)C)=O)cc2cc[nH]c2cn1 86185,C1(NC(C(CC)(C)F)=O)COC2(C1)CN(C(=O)C(C)(C)C(=O)OC(C)(C)C)C2 86186,C1(C(=O)NCc2ncc(C(N3CC(OC)(CO)C3)=O)cn2)CCOCC1(C)C 86187,N1(C(c2ncc(OC)cn2)=O)CCC2(C1)CN(C(c1cc(Cl)c(Cl)s1)=O)C2 86188,c1(OC)ccc(F)c(NC(=O)C(C)(CSC)NC(=O)CC(C)C)n1 86189,C1(CC(=O)NCC2CC(NC(=O)Cn3cnnc3)C2)CC2(CCC2)CCO1 86190,Cc1cc(C(N2CC(O)(C(C)NC(=O)CC(c3ccccc3)N(C)C)C2)=O)co1 86191,N1(C(C2(C)CC2)=O)CC2(CCN(C(C3(c4cccnc4)CCCCC3)=O)CC2)C1 86192,c1(OC)ccc(CNc2cccnc2C(N2CCc3sccc3C2)=O)c(F)c1F 86193,C1(CCNC(c2n(C=C)nnc2)=O)CCCN(C(=O)C(F)CC2CCOC2)CC1 86194,C1(NC(c2cc(OC)ncc2)=O)(CNC(c2ccc(Cl)cc2)=O)CCCCC1C 86195,C1(CNC(c2c(C)cc(SC)o2)=O)CN(C(=O)CN2CCCCC2C)CC1(F)F 86196,N1(C(CC(CC)SC)=O)C2CC=C(C(=O)NCC3C(C)C3(F)F)C1CC2 86197,N1(C(C(C(C)C)CO)=O)CC2(CCC2)CC1CNC(=O)COC1(C)CCOCC1 86198,c1(CN(C)C(C2COCC2(C)C)=O)cncc(O)c1 86199,C12(CNC(C3(CCCC)CC3)=O)CCC1CN(C(=O)C=Cc1ccc(C)s1)C2 86200,N(C(=NCC1C(C)C1C)NCC1CCOC1)CC1(OC)CCC1 86201,C1(F)(C(=O)NCc2occ(C(=O)NC(CCC=C)C)n2)CCCCC1 86202,c1(C(=O)NCC(C)NC(=O)C=CCOC2CCOCC2)cccc(C#N)n1 86203,CC(CC(=O)NCC1(F)CN(C(C2(F)CCOC2)=O)C1)c1ccncc1 86204,CCCCCCCCCC(=O)N1CC(C)(NC(=O)C(c2ccccn2)O)C1 86205,N1(C(=O)NC)CCN(C(C2(Nc3ccc(-c4nn[nH]n4)cc3)CC(F)(F)C2)=O)CC1 86206,C1(C(=O)NCC(C2CN(C(CCCN=[N+]=[N-])=O)C2)OC)CCCCC1CO 86207,C1(CNC(c2cnnc(O)c2)=O)CCN(C(c2ccccn2)=O)CC1O 86208,Cc1ccc(COCCN2CC(CCCNC(=O)C(C)(C)C3CCCO3)C2)cn1 86209,C(=O)(C(C)C(CC)CC)NC1C(NC(c2c(CC)n[nH]c2)=O)CC1 86210,N1(C(c2c(C)nc(C)s2)=O)CC(NC(=O)COCC(F)F)C(C2CC2)C1 86211,c1(N(CCNC(=O)C(C)CC2CCC2)CC)ccc(F)cc1C#N 86212,C1(NC(c2nc(C(C)C)sc2)=O)CCCC1(C)NC(=O)C(C)C1CC1 86213,c1(C(=O)NCC2CC(O)(CNC(C3(COC)C=CCC3)=O)C2)ccc(C)nc1C 86214,Cc1[nH]c(=N)nc(O)c1CCC(=O)NCC1CN(C(=O)CCC2CCCCO2)C1 86215,c1(C(N2CC3N(C(CCOc4cccc(C)c4)=O)C3C2)=O)c(Cl)cc(Br)cc1Cl 86216,C1(N2C(C(=O)NCc3ccn(C)n3)CCC2)CCN(C(c2ncccn2)=O)CC1 86217,n1(C(C)C)cnc(C(=O)NC(C)(C)CNC(=O)Cc2cncs2)c1 86218,N1(C(c2n(C(CC)CC)ncc2)=O)CCCC(N(C(C2CC3CC3C2)=O)CC)C1 86219,N1(C(C2C(C)C2C)=O)CCN(C(=O)C(Cl)=CCl)CCC1C 86220,C1(NC(=O)C(F)Br)CN(C(c2n[nH]c3c(F)cccc23)=O)C2(CCOC2)C1 86221,N1(C(C(CSC)C)=O)CCN(C(C2CC(n3cnnc3)C2)=O)CC1C 86222,C(C(C)(C)CC(=O)N1CCCC(CC(N)=O)C1)NC(C=CC)=O 86223,C(CCCC#N)(c1nnnn1C1CC1)NC(c1ccc(N2CCCCC2)cc1)C 86224,N=c1nc2c(C(N3CCCC3C3(NC(=O)Cn4cccn4)CC3)=O)cccn2[nH]1 86225,N1(C(Cc2c(COC)cccc2)=O)CCN(C(=O)C2=NOCC2)C2CC12 86226,C12(C(=O)NCC(C)(O)CCO)CCC1CN(C(=O)CCOCC(F)F)C2 86227,CCCC(CNC(C1CSCCN1C(c1cocn1)=O)=O)CCO 86228,c1(C(=O)NC2CN(C(CC(C)OC)=O)C2)sc2nccnc2c1N 86229,C=CCC(CNC(=O)COC1CC1(F)F)C(=O)N(C)Cc1nc[nH]n1 86230,N1(C(C(CC)N(C)C)=O)CC(NC(c2ccnc(OC)c2)=O)C2CCCCC12 86231,N1(C(c2c(C)cco2)=O)CCC(N=[N+]=[N-])(C(=O)N(C)CC2CC2(C)C)C1 86232,c1(NC(C(C2CCC2)NC(c2cc(COC)[nH]n2)=O)=O)cncc(SC)c1 86233,C12(C(=O)Nc3cccc(C)c3)CCCC1CCN2C(=O)C(C)Oc1ccccn1 86234,CCN=C(NCCCC(C)(F)F)NCCC1CCCC1(C)C 86235,Cc1ccc(C(=O)NC(CC(=O)NCc2c(F)cncc2F)C(C)C)c(C)n1 86236,C1(CNC(=O)C2=CCCS2)CCC2(CO1)CC(NC(=O)COc1ccccc1)C2 86237,N1(C(c2cnc(C(C)C)nc2)C(=O)Nc2c(C)cccc2)CC2CC3CC2C1C3 86238,c1(C(N2C(C)CC2C(=O)N(CCF)C2CC2)=O)cc[nH]c(=N)n1 86239,c1(OC)ccc(C(N)=O)cc1C(=O)NCC(C)(C)NC(=O)C=CCO 86240,Cc1cc(C(=O)NC(C2CCCCC2)CNC(C2CC(=O)N2)=O)ccc1[N+](=O)[O-] 86241,c1(OC)ccc(C=CC(=O)NC2(C)CCN(C(=O)C(C)C(C)(C)C)C2)cc1F 86242,c1(C(N2CCCCC(NC(C3C(C)C3)=O)C2)=O)cccnc1S(=O)(=O)C(F)(F)F 86243,c1(CC)ncccc1C(=O)N(C1CCC(NC(c2cccnc2)=O)C1)C 86244,c1(CC)ncc(C(=O)NC2CC(NC(C3(SC)CC3)=O)C23CCC3)c(O)n1 86245,c1(C(N2C(CNC(CCSCCCC)=O)CC(C)CC2)=O)ccn2ccccc12 86246,c1(C(=O)NCCNC(c2c(C)ccc(Br)c2)=O)coc2c(C)cccc12 86247,C=C(C)CC(C(=O)N(C1CCCN(C)C1)C)NC(c1cc(OC)ccn1)=O 86248,CC1CC(NC(c2cccc(=O)o2)=O)CN1C(=O)Cc1ccccc1Br 86249,N1(C(COCCOCC#C)=O)CC(NC(c2c(N)cccc2F)=O)CC(O)C1 86250,Cc1ccc2sc(C(N3CCC(O)(CNC(=O)C(C)CC(F)F)C3)=O)cc2c1 86251,c1(C(N2CC3C(CNC(CC(C)(C)C4CC4)=O)(C3)C2)=O)cc(O)ccc1Cl 86252,S(=O)(=O)(c1cnc(NCC23CCCC2OCC3)c(Cl)c1)NCCCN(CC)CC 86253,c1(C(=O)NC2CCN(C(CC3(OC)CCCC3)=O)CC2F)cccn2nncc12 86254,c1(C(=O)NCCC(C)NC(C(CCC)O)=O)c[nH]ccc1=NC(=O)C(C)(C)C 86255,CC(F)(F)CC(=O)N1CC(NC(c2ccncc2F)=O)C1 86256,CC1(NC(c2coc(Br)n2)=O)CCN(C(=O)CCCn2ccccc2=O)C1 86257,N1(C(CCC(=O)OCC)=O)CCC(CO)C(NC(=O)CCCn2ccnn2)C1 86258,N1(C(C(CC)O)=O)CC2CC3CC2C1C3NC(=O)CCc1cscn1 86259,N1(C(C=C(C)Cl)=O)CC(NC(=O)C(c2ccnn2C)O)C(O)C1 86260,N(C(=NCCC1CS(=O)(=O)C1)NCc1noc(C2CC2)n1)CC1CC(C)C1 86261,c1(C(=O)NC(CNC(c2c(OCC)oc(C)n2)=O)C2CCC2)cc(C)cc(C)c1 86262,N1(C(C(C=C)(C)O)=O)CC2CC(NC(c3ccc(CC)c(Br)c3)=O)C1C2 86263,C1(C(=O)O)CCCC(CNC(c2occc2-c2ccccc2)=O)C1 86264,c1(C(=O)NC2C(CNC(c3cccc(C(=O)NC)c3)=O)C2)ccc(Cl)c(N)c1Cl 86265,N(C(=NCCF)NCCc1cc(Cl)ccc1Br)CC1CCN(C)CC1 86266,c1(N(CCCNC(=O)CC(C)C2CCCO2)CC)ncncc1OC 86267,CC(C)(CCCNC(=O)CC(F)(F)F)C(=O)NCC1CCC(F)C1 86268,c1(OC)cc(C(=O)NCCNC(C23CCN(CC2)CC3)=O)cc(F)c1 86269,c1(N2CCC(CSC)C2)nccc(=NC(C)COC2CCCC2)[nH]1 86270,N1(C(=O)NCC2(C)COC2)CCC(O)(C(F)(F)C(N)=O)C1 86271,CN(Cc1cc(-c2cccc(Br)c2)no1)N1CC(C2(C)CCCO2)C1 86272,N1(C(C2C(COC)CC2)=O)CC2CC2(NC(C2CC(C(C)C)C2)=O)C1 86273,c1(C(N2C(C)C(=O)NCC2)C(=O)NCc2ccco2)cc2ccccn2n1 86274,N(C(=NCCCC(C)(F)F)NC(C)C1CC1)C(c1cccnc1)C 86275,C1(CC(=O)NC(C=C)(C)C)CN(C(C2CC3CC2CC3O)=O)CCC1C 86276,c1(OC)cc(Cc2nc(C(N)CC(F)F)n(-c3c(F)cccc3Cl)n2)ccc1C 86277,C(CCCCNC(CC)CSc1cccc(C)c1)(c1nnnn1C)SC 86278,FC1(F)CCC2C(CCCN2CC2CCc3cccnc32)C1 86279,c1(-n2cc(CC(CC(=O)OCC)N)nn2)cccc2ccsc12 86280,C(=O)(C1=COc2ccccc2O1)N(C1C2CN(C(C3CCC(C)(C)O3)=O)CC12)C 86281,N1(C(CN2C(C)CCC2)=O)CCC(CNC(=O)C=CC(c2ccc(F)cc2)=O)CC1 86282,c1(C(N2CC(C(C)NC(C3(CC=C)CC3)=O)OCC2)=O)cc2c(cn1)OCCO2 86283,C=C(Br)CCC(=O)NC1CCC(CNC(c2ccc(C(F)F)nc2)=O)C1 86284,Cc1c(O)c(=O)ccn1CC(N1CC2CC(NC(=O)C(F)C3CC3)C1C2)=O 86285,c1(C(=O)NCCC2CC(NC(C3C(C(C)=O)C3)=O)C2)c(C(N)=O)cnn1C 86286,Cn1c(O)ncc(C(=O)NC2CC2NC(=O)CC2CC3(COC3)C2)c1=O 86287,C(CC(C(C)(C)C)NC(=O)C(C)OC1CCOC1)N(C(c1c(C)noc1N)=O)C 86288,CC(C)(CC(=O)N1CC(NC(C2CCCCN2N=O)=O)CC(F)C1)CC(F)F 86289,C1(NC(C(C)O)=O)CC2(C1)CC(NC(c1c[nH]cc(F)c1=O)=O)C2 86290,c1(C(N(CCCNC(C2CCC=CCC2)=O)CCO)=O)ccnnc1S 86291,C1(NC(C(CCC)F)=O)Cc2ccccc2C1NC(=O)CC1C=CCC1 86292,CC(Cc1c[nH]c2ccccc12)N=c1[nH]c(=NCCC2CCC2)c2sccc2[nH]1 86293,N1(C(c2cnc(OCC)nc2)C(=O)NC(C)(C)C)CCN(C)C(CC)C1 86294,c1(NCC2OCC(CNC(=O)CC34CCC(CC3)CC4)C2)ncnc2sccc12 86295,c1(C(=O)NC2C(NC(Cn3ncn(C)c3=O)=O)CCC2)c(N)cccc1[N+](=O)[O-] 86296,C(C(C(=O)NCC1CC(O)CN1C(c1ccc2c[nH]nc2n1)=O)C(F)(F)F)OC 86297,c1(C(N(C2C(C)CCN(C(=O)CC3(C)CC3)C2)C)=O)ccc(Cl)c2ccccc12 86298,C1(NCCC(C)(C)OC)CCC2CN(C(=O)CCC=CC)CC2C1 86299,C#CC1CN(C(=O)CCc2nncn2C)CCN1C(=O)COCCN(C)C 86300,N1(C(C2(C(=O)OCC)CC2)=O)CC(C(=O)NC2CCCC(C)C2C)C(C)(C)C1 86301,C1(C(C)NC(=O)C(=O)NCC2(Cc3ccccc3)CCOC2)CC2CCC(C1)C2 86302,N1(C(c2cnc(C)o2)=O)CC=CCC1C(=O)NC(C)C1CC1 86303,c1(CC(=O)N(C)CC2CCCN2C(=O)CN2CCOC2=O)c(F)cccc1Cl 86304,c1(OC)ccc(C(=O)NCCC2CCN(C(C3(C(C)C)CC3)=O)CC2)nc1 86305,C(=O)(C1=CCCOCC1)N1CCC(CCOC)(NC(C2C(C)(CC)C2)=O)CC1 86306,C1(CNC(C(N2CCCCC2)C)=O)N(C(=O)CSc2n[nH]c(O)n2)CCC1(C)C 86307,C(=O)(C1=NNC(=O)CC1)NC(CC)(C)CCNC(c1ccn(C)n1)=O 86308,N1(C(c2cc(COC)on2)=O)CCC2CN(C(C3CC3c3ccsc3)=O)CC2C1 86309,N1(C(c2c(CC)n(CC)nn2)=O)CC(O)(C2(CNC(C3CC(C)CO3)=O)CC2)C1 86310,c1(CC(N2C(CN(C(CN(CC)CC)=O)CC)COCC2)=O)cc(C)ccc1O 86311,CC(C)C(C(c1ccccc1)NC(c1ocnc1CO)=O)NC(=O)OC(C)(C)C 86312,C1(C(=O)NCCN(CCOC)C(c2cnc(C)o2)=O)CCc2nnn(C)c2C1 86313,c1(C(N(C2CCN(C(=O)C(C#N)CC)C2)CC#C)=O)cn(C)nc1CC 86314,C1(C)(C(N2CCC(N(C)C)CC2)=O)CCCN(Cc2sccc2Br)C1 86315,C1(C(=O)NCC(C)CN(C(=O)C(C)c2ccco2)C)CCC2(CCCCC2)CC1 86316,Cc1cccc(C)c1C(C(=O)O)NCc1cc(Br)sn1 86317,N1(C(C(C)(C)OCC)=O)CCC2CCCC(C1)N2C(c1cc2c(nn1)CCC2)=O 86318,c1(C(=O)NC(CC=C)CNC(c2cc3scnc3[nH]2)=O)cc(F)c(F)cc1F 86319,N1(C(C(COC)OC)=O)CC(C(=O)N(CCCO)C(C)C)C(C)C1 86320,C1(CN(C(CN(CCC)C(c2ccc(C#N)o2)=O)=O)C)C(C)(C)C1(C)C 86321,N1(C(=O)CC2CCCC23CC3)CC=C(C(=O)N2CC(OCCF)C2)CC1 86322,c1(C(N2C(CC)CN(C(=O)C3=NNC(=O)C3)CC2)=O)cc2n(n1)CCCC2=O 86323,c1(C(=O)NCC2(NC(C3CCS(=O)CC3)=O)CCC2)ccc(F)cc1[N+](=O)[O-] 86324,C12(CNC(C(CCC)C#N)=O)CN(C(c3c[nH]nc3C(F)F)=O)CC1CCO2 86325,Cc1nc2cncc(C(N3CC4(CCN(C(c5c[nH]cc5Br)=O)C4)C3)=O)c2[nH]1 86326,CC(C)CCCCNC(c1ccn(CCNC(C2CC3(CC3)C2)=O)c1)=O 86327,C1(NC(CC2(OC)CCCC2)=O)COCCC1NC(C1CCC(C(C)C)CC1)=O 86328,c1(C(=O)NC(CC(C)NC(C2C(C)C2)=O)C)n[nH]c2c1CC(C)CC2 86329,C(CNC(=O)CCC1CC1C)(C(C)(C)C)NC(c1cc(CCCCC)[nH]n1)=O 86330,c1(OC)cc2c(nc1N1CCCC1c1nn(-c3ccccc3)cc1F)CCC2 86331,C=CC(C)CC(=O)NC1CC(CNC(c2ccccc2OC(F)(F)F)=O)C1 86332,c1(NC)cc(C(=O)NCCCCCNC(=N)N)ccc1F 86333,Cc1cc(C(=O)N(C2CCN(C(=O)COCC3(F)CC3)CC2C)C)ncc1C#N 86334,N1(CCOC)CC(NC(=O)C(C)OC2CCCC2)CC1=O.C12CC(C1)C(=O)N2 86335,N1(C(c2nnc(-c3ncccc3Cl)s2)=O)CCC2(CCNC2=O)C1 86336,c1(C(N2CC(NC(c3ccnc(C)c3O)=O)C(C)C2)=O)cc2c(C)n[nH]c2cn1 86337,c1(C(=O)NC(CC)(C)CNC(=O)C#CC(=O)N(C)C)n[nH]c2ccc(O)cc12 86338,N1(C(C(COC)OC)=O)CCOCC(NC(=O)CCCCCO)C1 86339,C1(O)(CC(=O)NCCCCNC(CSc2nc(C)[nH]n2)=O)CCCOC1 86340,Cc1ccc2c(C(=O)NCCCNC(=O)C(F)=CCCF)cnn2c1C 86341,CC1CC(C(N2CCOC(C(N)=O)C2)=O)N(C(=O)CCC2(C#N)CCC2)C1 86342,C=CC1(CC(=O)Nc2c[nH]ccc2=O)CN(C(=O)COCCC)C1 86343,c1(N2CCCCC(NC(CC(=C)C)=O)C2)nccc(S(C)(=O)=O)n1 86344,c1(C(N2CCCC(C(C)NC(C(C)=CC)=O)C2)=O)cccc2[nH]c(=N)oc12 86345,N1(C(C(CC2CCC2)OC)=O)CCCC(N(C(=O)Cc2cnoc2)C)C1 86346,C1(CNC(CC=C)=O)CCN(C(=O)CCc2nc3ccccc3o2)C12CCC2 86347,C(=O)(CC(C)(C)C=C)NCC(=C)CCNC(=O)CC(CC)c1ccccc1 86348,N1(C(C(C(=O)OCC)(C)C)=O)CCc2sc(CNC(=O)CS(N)(=O)=O)nc2C1 86349,N1(C(=O)OC(C)(C)C)CC2(CCCN(Cc3ccc(F)c(O)c3)C2)C1 86350,C1(CCC(=O)N(CC)Cc2cnn(C)c2)CCCCN1C(C1C=CCCC1)=O 86351,c1(C(=O)OCC)nn(C)[nH]c1=NC(=O)c1noc(C)c1Br 86352,N1(CC)C(=O)CCC1CC(N1CC(CNC(c2c(C)nsc2N)=O)C1)=O 86353,CC1(C)NC(=O)CCC1C(S12C(CC(F)(F)C1)COC(=O)N2)=O.C(C)(C)(C)O 86354,C1(NC(=O)C=CC2CCC2)CCC12CN(C(C1CCN(C3CC3)C1=O)=O)C2 86355,C=CC(O)C(=O)NCC1CCC(NC(=O)CN(C(=O)COC)C)C1 86356,O=C(CCC(CF)CF)NCC(C1CC1)NC(=O)CCc1ccc(F)cc1 86357,N1(C(C=C(C)c2ccco2)=O)C(CC(=O)NC2CCCC2O)C2CCCC12 86358,c1(C(N2C(C)C(NC(=O)Cn3cccnc3=O)CC2)=O)cccc(S(N)(=O)=O)c1 86359,C1(C(N(CCN(C(c2cc(C(C)(C)C)on2)=O)CC)CC)=O)CCc2nnnn2C1 86360,CC1CN(C(=O)Cc2n[nH]cc2Br)CC1CNC(=O)CCc1cncn1C 86361,c1(C(=O)NC2C(C)N(C(=O)CC3CCC4CC34)CCC2)cn2cc(Cl)cnc2n1 86362,c1(C(=O)NCC2CC(OC)CN2C(=O)CNC(=O)C2CC2)cc(C)n(C)c1C 86363,c1(-c2c(OCCOC)cccc2)nc2c(C(=O)O)ccc(Br)c2s1 86364,C(=O)(CCCC(=O)OC(C)(C)C)NC(CNC(C1CN(C(C)C)C1)=O)(C)CO 86365,C1(C(=O)NC(C2(O)CN(C(C3(OCC)CCCC3)=O)C2)C)CCOC(C)(C)C1 86366,CCC(F)(F)CC(=O)N(C)CC1CCCC(NC(=O)CCc2ccoc2)C1 86367,c1(C(=O)NC2CCN(C(=O)C=Cc3ncc[nH]3)CC2F)cnn2ccc(O)nc12 86368,c1(NC(C2CC3CC3N2C(=O)CC2CCCCO2)=O)ncc(Br)nc1Br 86369,Cc1cc(=NCCN2CCC(N(C)C)C2)[nH]c(NC2CCC3(C(C)C)CC23)n1 86370,c1(C(=O)OC)cc(C(C)=O)ncc1OCc1nc(Cc2ccccc2F)no1 86371,c1(N2CCC(NC(c3cn(CCCC)nc3C)=O)C2)ccc(C#N)nc1 86372,C1(CC(=O)NC(C2CCCN2C(c2c[nH]nc2C(F)F)=O)(C)C)CCC2CC2C1 86373,C1(NC(c2cc[nH]n2)=O)CCCC(NC(C23CSC(C2)C3)=O)C1 86374,N1(C(CC2COCC(C)(C)O2)=O)CCc2ccccc2C(NC(C2COC2)=O)C1 86375,c1(NC(=O)NC2CC(c3ccc(Cl)cc3)C2)ccc2nc(O)sc2c1 86376,CC1NC(=O)C(C)N(Cc2ncc(C(F)F)cc2Cl)C1C 86377,c1(NC(=O)NCC2CCCN(CC(F)(F)F)C2)snc(-c2ccccc2)c1C#N 86378,N1(C(CCN(C(C(C)C)=O)CCO)=O)CCCCC(CC(C)C)C1 86379,C#Cc1ccc(C(=O)NCC(C)(C)CNC(c2c[nH]cc2C2CC2)=O)nc1 86380,N1(C(C(C)NC(C)=O)=O)CCCC(CCNC(c2conc2C(C)(C)C)=O)CC1 86381,Cn1cc2ncc(C(N3CCN(C(=O)CC4CCCO4)CC3)=O)cc2n1 86382,C1(c2n(C)cnc2)CN(C(C2(C)CNC(=O)C2)=O)CC1NC(=O)C=CC(F)(F)F 86383,c1(C(N2CCC(OC)C2)C(=O)NCCSC2CCOCC2)ncc(C)cc1C 86384,Cc1noc(C(=O)NC(Cc2ccccc2)C(=O)O)n1 86385,CN1CC2CCC(C1)N2C(C1CCN1C(c1cc(-c2ccncc2)no1)=O)=O 86386,C(C(C(=O)NCC(CC)NC(=O)C=Cc1cccs1)c1ccccc1)OCC=C 86387,C12(NC(=O)Cn3ncc4ncccc34)CC3CCC(C1C2)N3C(C1C=CCC1)=O 86388,C(CC(O)C(=O)NCc1cn(CC(=O)NC(c2cccnc2)C)nn1)SC 86389,C(=O)(C1CCCc2scnc21)NCC(C)(C)Nc1nc(Cl)nc2c1CCC2 86390,N1(c2nnc(CCC)s2)CCN(C(c2ccc(CCC)[nH]2)=O)CC(C)(F)C1 86391,CCCC(C(O)C(=O)N1CC(N2C(=O)CCC2=O)C1)NC(C12CCCC1CCC2)=O 86392,N1(C(c2cc(CC)[nH]n2)=O)CCOC(CN(C)C(C2CCCN(C(N)=O)C2)=O)C1 86393,C1(C(C)NC(=O)Cn2ccc(C)c2)CN(C(=O)CC2CCC2)CCO1 86394,Cc1cc(CNC(C2CC(C)CN(C(c3c[nH][nH]c3=N)=O)C2)=O)cc(F)c1 86395,N1(CC)C(C)CN(Cc2c(OC)nsc2OC(C)C)CC1(C)C 86396,CCCC(CNC(c1cc[nH]n1)=O)C(=O)N1CCCC1C1(CO)CC1 86397,N1(C(C2C(C(C)C)CN(C(C3CC(C(C)C)C3)=O)C2)=O)CCn2nccc2C1 86398,c1(C(N2C(CNC(=O)CCC(C)C)CC(OC)C2)=O)nccc2c(F)cccc12 86399,C1(C2CCCC2)(C(=O)NCc2ccc(CNC(C34CC(F)(C3)C4)=O)cc2F)CCC1 86400,c1(CN2CCC(C)C(C)(C)C2)ccc2cc(F)cc(Br)c2n1 86401,c1(C(=O)Nc2c(OCC)cc(Cl)cc2)ccc2[nH]nc(Br)c2c1 86402,N1(C(c2ccc(F)c(Br)c2F)=O)CCOC2CCNCC12 86403,Cc1nn(C)c(=O)c(C(N2CC(F)(CNC(=O)C(n3cc(Cl)cn3)C)C2)=O)c1C 86404,Cc1c(C(=O)NC(CNC(c2ccsn2)=O)CO)cnc2ncnn12 86405,C1(NC(C(C)O)=O)C=CC(CNC(=O)C(C)(C)c2cncnc2)C1 86406,c1(C(N2CC(NC(C(C(C)C)n3ccc(C)c3)=O)C2)=O)cnn2c1OCCC2 86407,c1(C(N2CC3CC2CN3Cc2cscc2Br)=O)cc2n(n1)CCC2 86408,C12(CCNC(C3C(C(=O)OCC)C3)=O)CCC1CN(C(=O)Cc1ncsc1Cl)C2 86409,CC(C)(CO)C(=O)NC1CC1NC(c1ncoc1C(C)(C)C)=O 86410,C=C(Cl)CC(C(=O)NC1CCC(=O)NC1)NC(=O)C(F)CCC 86411,Cc1c(C(=O)NC(C)C(CO)NC(C2(C)CC(C)C2)=O)cnn1C(C)C 86412,C1(NC(c2c(C)n(C3CCC3)nc2)=O)CC2(CCN(c3ccnc(C#N)n3)C2)C1 86413,Cc1nc(NCCc2nnc3n2CCS3)cc(=NC(C)c2cc[nH]n2)[nH]1 86414,Cc1cccc(C(F)C(N2CC(C)(NC(c3cncc(N(C)C)c3)=O)C2)=O)c1 86415,N1(C(C(C(C)(C)C)O)=O)CCN(C(=O)CC2=NNC(=O)C2)C2COCC12 86416,c1(COC(=O)CC2CC2(Cl)Cl)c2c(coc1=O)CCCC2 86417,N1(C(C2N(CC)CCC2)=O)C2CCC1CC(C(=O)NCC(F)C1CCC1)C2 86418,c1(C(=O)NCC2(OC)CN(C(c3cncc(C)n3)=O)C2)c[nH]nc1[N+](=O)[O-] 86419,C12(C(N(C(C)C)C)=O)CC1CN(C(=O)CN1CCN(S(C)(=O)=O)CC1)C2 86420,Cc1nncn1NC(=O)C1CC(NC(c2csc(F)c2)=O)CCO1 86421,CC1CCN(C(c2csnn2)=O)CCC1N1CCCC1c1c(F)cccc1Cl 86422,c1(C(C)=O)cc(C(=O)NC(C2CCN(C(=O)C(C(C)C)NC(N)=O)C2)C)c(C)o1 86423,C1(C(N(CC(C)NC(c2ccncn2)=O)C)=O)C(C)CCN1C(=O)OC(C)(C)C 86424,C(=O)(CC1=CCN(C(C2CCOC2(C)C)=O)CC1)NC1(C)C(C)C1 86425,N1(C(c2cc(CC)c(F)cc2)C(=O)NC(C)C)C2C=CCC1CCC2 86426,c1(C(N(C2CN(C(C3CC34CC(O)C4)=O)C2)C)=O)ccnc(F)c1 86427,c1(C(N2CCC(CCC(=O)N(C(C#C)C)CCCC)C2)=O)cc(C#C)ccn1 86428,c1(N(C)C)[nH]c(=NCC2(C(=O)NOCC=CCl)CCCC2)nc2sccc12 86429,CCCC(C(O)C(=O)NC1CCN(CCCO)C1)NC(=O)CC(C)(C)COCC 86430,CN1CCC(C(=O)NC2CCN(C(c3cccc(NS(C)(=O)=O)c3)=O)C2)C1=O 86431,c1(C(N(C)CCOCCNC(=O)Cn2cnnc2O)=O)cn2ccsc2n1 86432,O=C1CS(=O)(=O)CC(C(=O)NCC2CC2NC(=O)C(F)F)N1 86433,c1(CC2(C(N(CC(C)NC(c3cnn(C)c3)=O)C)=O)CCCC2)ccc(Cl)nc1 86434,N1(C(C(CCC)OCC)=O)CC2(C(=O)NCC(CO)C3CCC3)CC1CO2 86435,Cc1cnc(C)c(NC(C2C=CCN2C(c2cccc(Cl)c2F)=O)=O)n1 86436,c1(C(=O)NCCOCCCC#C)ccnc(CNC(C2(C)CC3CC3C2)=O)c1 86437,N1(C(C(C)C)=O)CC(CNC(C2NC(=O)CC2C(F)(F)F)=O)C(C)C1 86438,C(=O)(C1=CCCN(Cc2cnccc2N(C)C)C1)Nc1ccc(OC)c(OC)c1 86439,c1(NC(c2c(CNC(CSCCC#N)=O)noc2)=O)cccc(F)c1 86440,C1(NC(c2c(C)cns2)=O)C(C)CCN(C(c2cnc3sccn23)=O)C1C 86441,c1(C(N2C(CNC(c3nc(C4CC4)cs3)=O)CC(O)C2)=O)cc(F)ccc1Cl 86442,C(C(C(=O)N1CCCC1CNC(c1cc(C)ns1)=O)C(C)(C)C)OCC=C 86443,C(=O)(C1=C(Cl)CCCC1)NCC(C(C(=O)NCC(=C)Cl)F)C 86444,N1(C(C)C)CCCCC1C(=O)NC1(C)CN(C(C2(S(C)(=O)=O)CC2)=O)C1 86445,CC(CN(C)C)CCC(=O)NCc1ccc(C(=O)NCC2C3CCCC23)s1 86446,N1(C(CCC)=O)CCCC(C(N2CC(O)(CNC(=O)CCC(N)=O)C2)=O)C1 86447,C(=O)(C1CCCc2scnc21)NCC(CC)NC(C1CCc2nncn2C1)=O 86448,c1(C(N2CCC(N(c3nccc(C#N)n3)C)C2)=O)ccc(C#N)c(F)c1F 86449,C1(NC(CSCCCC)=O)CCCN(C(=O)CCc2ccoc2)C1C 86450,N1(C(C(C(C)(C)C)=O)=O)CCC(C(N2CC3C=CCC(C3)C2)=O)C(C)(C)C1 86451,Cc1noc(C)c1-c1cn(C2CCCC2NC(C2(C(F)F)CC(O)C2)=O)nn1 86452,N1(CCNC(C2(CCNC(C3(CC)CCC3)=O)CC2)=O)CCNC(=O)C1 86453,c1(-n2cc(CC(C(=O)NCCN(C(=O)OC)C)O)nn2)cccc(C(=O)O)c1 86454,CC1(CCCCNC(N2CCCC2c2ccc(Cl)nc2)=O)NC(=O)NC1=O 86455,Cc1c(C(=O)NCCCCCN(C)C(c2cncc(C(C)C)c2)=O)ncn1C 86456,c1(C(=O)NCCNC(C2CCCOC2)=O)ccc2c(Br)cccc2c1 86457,C1(NC(C(C)OCCN(C)C)=O)CCCC1CNC(C1(F)CC1)=O 86458,c1(C(=O)NC2C(NC(C3C(C(C)C)C3)=O)CCC2)nc(-c2ccccc2)sc1N 86459,CCC(CNC(C1CN(C(N)=O)C1)=O)(CC)NC(C1CCNC1=O)=O 86460,C1(CNC(CCNC(COC)=O)=O)CC(C)(C)CN1C(c1cscc1COC)=O 86461,c1(C(N(C2C(C)CCN(C(=O)C(O)C3CCC3)C2)C)=O)cc2ncccc2[nH]1 86462,c12nc(cn3ccnc13)N1C(COC)CN2CC1.c1(C(=O)N(C)C)ccccc1 86463,c1(C(=O)NCC2(C)CCCN2c2cc(Cl)ncn2)cnc2cnccc2c1 86464,c1(C(=O)NC(C)CNC(c2ccncc2N)=O)cc2nccc(C(F)(F)F)n2n1 86465,C1(NC(C(C)OCC=C)=O)CCS(=O)(=O)C12CN(C(=O)CSCC#N)C2 86466,N1(CC(=O)NC2CC(CNC(C(C(C)C)F)=O)C2)CCc2ccccc2C1=O 86467,C(=O)(CCS(=O)(=O)CC(C)C)N1CC(NC(C2=C(C)S(=O)(=O)CC2)=O)C(C)C1 86468,Cc1cc(C(N2CCOCC(NC(c3ncc(Cl)s3)=O)C2)=O)c(N)c(Cl)c1 86469,C(=O)(C(F)(F)CCNC(C1CCS(=O)(=O)N1C)=O)OCC 86470,C1(C(C)NC(C2(C(F)F)CC(=C)C2)=O)CCN(C(C2(C)CCCOC2)=O)CC1 86471,C(=O)(C1=CC(O)CCC1)NCC1CC(OC)CN1C(c1ccsc1Cl)=O 86472,n1(CC)nc(C)c(C(=O)NC2CCCCC2CNC(c2cc(F)n[nH]2)=O)c1Cl 86473,c1(C(=O)OC(c2ccc(Br)nc2)C)cc2c(C(F)(F)F)cc(N)cc2s1 86474,c1(CC)sc(C(=O)NCC(C)(C2CC2)NC(=O)C(C2CCC(=O)N2)C)cc1C 86475,N1(Cc2nc(C(C)SC)nn2-c2ccc(C)c(F)c2)CCC(C23CC(C2)C3)C1 86476,CC1Cc2cccc(C(=O)NC3CC(NCc4ccc5ncccc5c4)C3)c2O1 86477,C1(CC(=O)N(CCCC(=O)NCC(O)COC2CC2)C)CCC(C)(C)C1 86478,c1(C(N2CCC(NC(C(CCC)C)=O)C2)=O)cc(OC(F)F)ccc1C 86479,N1(C(c2cc(NC(C)=O)ncc2)=O)CCN(C(C2(C)CCCCC2)=O)CC1C#N 86480,c1(C(=O)NCC23CC(C(=O)NC4(C)CCCS4)(C2)C3)ccc(C#N)c(F)c1 86481,C1(N(C(=O)CC2CN(C(C)=O)CCO2)CC)CCN(C(c2cnc(Cl)[nH]2)=O)CC1 86482,C1(C(N2CC(O)(C(C)NC(c3c(OC)c[nH]n3)=O)C2)=O)C2CCCCC12 86483,c1(C(=O)NC(C2CCN(C(C=C(C)C(C)(C)C)=O)CC2)C)c(F)ccnc1Cl 86484,CC1(C)CC(CNC(c2cnc(C(N)=O)s2)=O)CN1C(c1cccc(F)c1)=O 86485,C(=O)(C(O)CC(C)(C)C)N1CC2C(NC(CCOC(C)C)=O)(C2)C1 86486,c1(C(N(CC(C)NC(=O)CCCCNC(N)=O)C)=O)ccc2cccc(F)c2n1 86487,c1(CC)ccc(C(=O)NCC2(NC(=O)Cc3c(C)nn(C)c3Cl)CCC2)cc1N 86488,N1(C(CSCCC(C)C)=O)CCC2CC1CN2C(=O)C(c1cncc(F)c1)C 86489,N1(C(C2(NC(=O)Cc3ccccc3O)C(C)(C)C2)=O)CC2(C)COCC2(C)C1 86490,C1(OC)CC(NC(C2CCCS2)=O)CN(C(c2cnn(C3CCC3)c2)=O)C1 86491,c1(C(=O)NC(CN(C(=O)C(C)Cc2ccco2)CC)C)ccsc1OC 86492,C1(C(C)C)CN(C(c2cc(N(C)C)ccc2F)=O)CCC1NC(C1CC=CC1)=O 86493,C(=O)(C(C)(O)C(C)(C)C)NCC(CNC(C1CC2(CC(=C)C2)C1)=O)O 86494,Cc1cc(C(=O)NCCCN(C)C(C2(C)CC(=O)N(C)C2)=O)cc(C(F)F)c1 86495,CC1(C)CCN(C(C2C3CCCOC23)=O)CC1NC(c1ccc(C2CC2)nc1)=O 86496,c1(C(N2CCC(C(CNC(CC(C)OC)=O)F)CC2)=O)cc(N)c(F)cn1 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86514,c1(C(=O)NCC2CCC(CNC(C(C)C(C)(F)F)=O)CC2)cccc2[nH]ccc12 86515,C1(C(C)NC(C(C2CCC2)OC)=O)CCN(C(C2(CO)CCCC2)=O)C1 86516,CN1CCC(NC(=O)CCN(C(=O)Cn2c(O)nnc2O)CCO)C(C)(C)C1 86517,c1(-c2nc(CCCC(=O)OC(CCC=C)C)on2)ccc(Cl)cc1 86518,c1(C(N2CC(C#C)N(C)CC2)=O)nn(CC)c2c1COCC2 86519,N1(C(c2c(CCC)nco2)=O)CC2CCC(C1)C2NC(=O)COC(C)C 86520,C1(NC(C2CC(=C)C2)=O)CCCC12CCN(C(c1cnc(OC)cc1F)=O)C2 86521,N(C1CCN(C(=O)OC(c2cc(Cl)cc(C)c2I)=O)c2ccc(Br)cc21)C(=O)NC(C)(C)C 86522,C1(CC(N2CCC(CN(C(=O)CSCc3ccccc3)C)C2)=O)NC(=O)NC1=O 86523,C(=O)(C(C(=O)N1CCC(C(C)(C)C)(CNC(=O)C(F)C(C)C)C1)OC)OC 86524,CCC1=NOC(C(=O)N(CC(C)NC(c2ccccc2CC(F)(F)F)=O)CC)C1 86525,CC(C)(C(=O)N1CCC(NC(C2CCOC2C(F)(F)F)=O)C1)c1ccsc1 86526,Cc1cc(=NCCNC(N2CCn3cc(C)nc3C2)=O)[nH]cn1 86527,C1(C(N(C)Cc2cccc(C)n2)=O)CCCCCCN1C(C1CC1C(N)=O)=O 86528,N(C(=NCc1cc(C2CC2)on1)NC1CC(=O)N(c2ccccc2)C1)C(C=C)C 86529,C(C(=O)N(C)O)N1CC1=O.C(C(=O)N(C)CCC1CCC1)N(C(=O)OC)C 86530,c1(CC)cccc(C(=O)N(CCCCCCNC(C23CCC2C3)=O)C)c1 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86549,CCC(C)(C(=O)NCC1CC(NC(=O)C(c2cccnc2F)(C)C)CC1O)OC 86550,n1(CCC(C)C)cc(C(=O)NCCCNC(=O)CC2(O)CC2)cn1 86551,C1(CCNC(C(=O)N(CCCS(=O)(=O)NC)C)=O)CC2(CCC2)CO1 86552,CCCC(CCC)=CC(N1CC(C(=O)N(C)Cc2cn(C)nn2)C(F)C1)=O 86553,c1(C(N2CC3C(CCNC(CCOCC#C)=O)(CC3)C2)=O)nc[nH]c2ncnc1-2 86554,C1(NC(C2CCS(=O)CC2)=O)C2CCC1N(C(=O)CC1=CCCC1)C2 86555,C#CC1(C)CCCN(C(=O)C(O)CCCNC(=O)C(C)(O)C=C)C1 86556,c1(C(N(CCCN(C(C(C)(CO)NC(C)=O)=O)C)C)=O)ccnc(F)c1N 86557,c1(C(N(CCCN(C(CSCC#C)=O)C)C)=O)ccc(C(C)=O)[nH]1 86558,c1(C(=O)NC2(C(=O)NC3CCC4(CCC4)C3)CC(F)(F)C2)c[nH]c2ncccc12 86559,n1(CC(=O)NCCC(O)CNC(C2CCCO2)=O)cc([N+](=O)[O-])c2ccccc12 86560,C#CC(C)(C)CCC(=O)Nc1ccc(Oc2ccc(F)c(Cl)c2)cc1 86561,C1(C)(CNC(=O)NC(C2CC3CCC2C3)C)CCN(C)CC1 86562,C1(NC(C(C)=C(CC)C)=O)CN(C(=O)COCC2CCC2)CCC1CO 86563,Cc1nc(=N)[nH]cc1C(N1CCC(N(C(=O)Cc2ccno2)C)C(C)C1)=O 86564,c1(C(N2C(CCNC(CC(=O)NCC#C)=O)CCCC2)=O)cnc2ccccn12 86565,N1(C(CSC)=O)CCCC(N2CCN(C(=O)CC3CCCC34CC4)CC2)C1 86566,C(=O)(CCCC(N)=O)NCC(C)CNC(=O)Cc1ccn(C)n1 86567,N1(S(CC)(=O)=O)CCC(C(=O)NCC(C)CNC(c2cnc(=N)[nH]c2)=O)CC1 86568,C(=O)(C1COc2ccc(Cl)cc21)NC(CC=C)CNC(c1ccsc1OC)=O 86569,N1(C(C2CCCN(C)C2)=O)CC(C2CCCN(C(c3cc(Cl)on3)=O)C2)C1 86570,c1(NC(c2c(F)ccc3c2OCO3)C)ccc2nc(N(C)C)[nH]c2c1 86571,C1(CC)CN(C(C2CC(F)C(=O)N2)=O)CCN1C(=O)Cc1cc(C)ccc1F 86572,O(NC(=O)C(C)(CSC)NC(=O)C(CC)N(C)C)CCCC#C 86573,c1(CC(=O)NCCN(CC(C)O)C(=O)C=CCF)cccc(C(C)(C)C)c1 86574,Cn1nc2c(c1C(=O)Nc1cnccc1Cl)CN(C(C1CCCCO1)=O)CC2 86575,CC(C)C1=NOC(C(=O)NCC=C2CCN(C(C3CC(C4CC4)C3)=O)CC2)C1 86576,c1(NC(C2C(NC(C(C)(C)OC)=O)C2)=O)cc(F)cnc1Br 86577,CCC(C(=O)NCC(C1CCC1)NC(=O)C=Cc1cocn1)n1cncn1 86578,C1(NC(c2ccc(C)cc2)=O)CN(CC23CC(C(F)F)(CO2)C3)CC1(C)C 86579,c1(C(=O)OC)c(C)[nH]c(C(=O)NC2CC2CNC(c2cc(C(N)=O)c[nH]2)=O)c1C 86580,C(=O)(C(C)CC(F)(F)F)NCC1COCCN(C(CCc2c(C)n(C)nc2)=O)C1 86581,N1(C(CC2CC(CC)OCC2)=O)CCOC2(C1)CN(C(=O)CC1C=CCCC1)C2 86582,Cc1c(CC(=O)NC(C)(CNC(c2cnn(CCO)c2N)=O)C(C)C)cnn1C 86583,c1(Nc2cccc(OCC(=O)NC(C)CCF)c2)ccc(S(N)(=O)=O)cc1 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86601,C(=O)(C(CCOC)OCC1CCC(C)C1)NCCNC(COCCCC)=O 86602,N1(C(C(CC)F)=O)CCC(O)(CNC(=O)CC(c2ccc(C)cc2)C)CC1 86603,C(=O)(C(C(F)(F)F)C(F)(F)F)NC1C(C)N(C(C2CN3CCCC3CO2)=O)CC1 86604,C1(NC(=O)Nc2c(C#N)nc(Cl)cc2)CC2(CCCCCCC2)C1 86605,C1(C)(NC(C(C)Cc2ccccc2)=O)CCC(NC(=O)COCC2(F)CC2)CC1 86606,C1(CNC(C2C(C)(C)C2)=O)CCC(F)(CNC(c2sccc2-n2ccnn2)=O)C1 86607,c1(-c2cnc(NC(c3nn(C(CC)C)c(C)c3)=O)s2)cccc(C#N)c1 86608,C1(CNC(CC=CC(C)(C)C)=O)CC(F)(F)CN1C(=O)C(O)Cc1ccccn1 86609,c1(N2CCC(COC(COCC(=O)OC(C)(C)C)=O)CC2)cc[nH]c(=N)n1 86610,Cc1nn(C(C)C)cc1C(N1CCC(CF)(NC(=O)COCC2CCCC2)C1)=O 86611,C1(CC(=O)NC2C(F)CCN(C(COC(C)C)=O)C2)CS(=O)(=O)CCN1C 86612,c1(NC(CCC2(NC(CCC)=O)CCC2)=O)c(C)ccn(C)c1=O 86613,N1(C(C(C)c2cccs2)=O)CC(C2CCCN(C(C3(C4CCC4)CCC3)=O)C2)C1 86614,c1(OC)ccc(NC(=O)CN(C)C(c2nc(C)ccc2C)=O)cc1F 86615,CON=CC(=O)N(CCCNC(C1CCC(C(C)(C)C)O1)=O)Cc1ccccc1 86616,C(=O)(CS(=O)(=O)C1CC1)NC1C(CC)CN(C(C2(F)CCN(C)CC2)=O)CC1 86617,CCCCCC(O)C(C)C(=O)NC1(CNC(=O)CCCCCC)CCOC1 86618,C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CC)(CNC(c1cnco1)=O)CC 86619,C(=O)(CC(=O)NC1CC1)NC(C1CCCN1C(c1csc(-c2ncc[nH]2)n1)=O)C 86620,CC(C)C(O)C(F)(F)C(=O)N1CC2CCN(C(=O)CCCC(C)(C)C)CC2C1 86621,C1(C(=O)NC2(CO)CN(C(C(CC#C)C3CC3)=O)C2)CC2(C1)CC2(F)F 86622,C1(C(=O)NCCCN(C(=O)Cc2cccs2)C)CCCC(N(C)C)C1 86623,CCC(CC(=O)NCC1(O)CCN(C(c2ncoc2Br)=O)C1)C1CCC1 86624,c1(CC)cc(C(=O)NC2CN(C(C3(CO)CC(C)(C)C3)=O)CC2OC)oc1CC 86625,C(=O)(C(CC)CC(F)(F)F)NCC1CN(C(CCCC)=O)CC(C)(C)C1 86626,c1(C(=O)NCCC2N(C(C(C=C)OC)=O)CCOC2)cc(C)c2occc2c1 86627,CCC(C(=O)NC(C)Cn1cc(C2CCCO2)nn1)N(C)C 86628,c1(C(=O)NCC2CCS2(=O)=O)ccc2c(c1)NC(=O)CCN2 86629,Cc1ccnc(CN(C)C(C2COCCC2NC(=O)C(C2CCCCC2)F)=O)c1 86630,c1(NCc2cc(NC(=O)C(F)(F)F)ncc2)cc(F)c(N2CCCC2)c(F)c1 86631,C1(NC(CCC(=O)NCC)=O)CN(C(c2ccc(N)c(F)c2)=O)CCC1(C)C 86632,c1(CCC(N2CC(CC=C)(NC(=O)C=C(C)CCC)C2)=O)cncc(OC)c1 86633,C1(NC(c2cnc(C)o2)=O)CCS(=O)(=O)C12CN(C(=O)CCS(C)=O)C2 86634,C1(NC(C2C(OC)C2)=O)CCCCC1C(=O)NCc1ccccc1OC(F)(F)F 86635,c1(C(N2CC(NC(CC(C)(C)C)=O)C3(C2)CC3)=O)cc2ccc(F)cc2[nH]1 86636,C=CCC(C)(C)CC(=O)N1CCC(C)CC1CNC(=O)CC1(N(C)C)CCC1 86637,c1(C(N2CCCC2CNC(C2CC(F)(CF)C2)=O)=O)ccc2c[nH]nc2n1 86638,c1(C(N2C(CNC(CS(CC)(=O)=O)=O)CC2)=O)cc(Cl)c(C)cc1[N+](=O)[O-] 86639,c1(C(=O)NCCCC(=O)NCCC2CC=CCC2)cc(O)ncc1F 86640,CC(C)CC(C)C(=O)NCC(C)(F)CNC(C1(CO)CCC1)=O 86641,Cc1cnc(C(=O)NC(C)(C)CN(C)C(c2ccc(C(C)(F)F)nc2)=O)cc1C 86642,N1(C(=O)OC)CSCC1C(N1CC(O)(C(C)NC(c2c[nH]cc2C(C)C)=O)C1)=O 86643,c1(CNCC(C)C(C)(C)C)cccnc1C(c1nnnn1C)OC 86644,C1(CNC(C(C(=C)C)(C)C)=O)CN(C(=O)CC2(O)COC(C)(C)C2)CCC12CCC2 86645,C1(c2nnnn2C2CC2)(NCc2ccncn2)CC2COC1C2 86646,C1(CNC(c2[nH]cc(C)c2)=O)(NC(=O)CCN(CC(F)(F)F)C)CCCCC1C 86647,C(=O)(C1CCCc2ncnn21)NCCCN(C)C(c1cc(Br)ccc1F)=O 86648,c1(OC)ncc(C(=O)NC2CC(F)(CNC(=O)CCCN(C)C(C)=O)C2)c(C)n1 86649,N(C(=NCC1CC1)NCC1(C)CCCC1)CC(C)(C)OC 86650,n1(CCC)nnc(=NC(=O)CC2CCNC2c2ccc(Br)c(C)c2)[nH]1 86651,c1(OCCC(N2CC(NC(CCC=CC(C)C)=O)C(F)C2)=O)ccc(C)cc1C 86652,c1(Cc2cn(C3CCN(C(C=COCC)=O)C3)nn2)c(Cl)cc(Br)cc1Cl 86653,c1(C(=O)NC2C=CCN(c3nnc(C4CC4)s3)C2)ccc2c(c1)CCCC2 86654,N1(C(C(N2CCOCC2)C)=O)CCOC(CNC(C2(N(C)C)CC(O)C2)=O)C1 86655,c1(CC)ncsc1C(=O)NC1(CNC(=O)C(F)CC2CC2)CC1 86656,c1(NCc2scc(CC(=O)OC)n2)nccc(=NC(C)c2ccccc2SC)[nH]1 86657,C1(NC(CC(C)(C)O)=O)CC2CC(C1)N(C(c1cnncc1C(F)(F)F)=O)C2 86658,CCCC(C(=O)OC)C(=O)N1CCCN(C(=O)Cn2cc(Cl)cn2)CC1C 86659,c1(C(=O)NCC(O)Cc2ccccc2Br)coc2c(Cl)cc(Br)cc12 86660,CC(CNC(=O)CN(C(c1cc(C#N)cs1)=O)C1CC1)CC(C)O 86661,C1(NC(=O)Cc2cccnc2O)CN(C(c2ccoc2)=O)CC2CCCC12 86662,c1(-c2cnc(OCC)nc2)nc(C(=O)Nc2ccc(C(=O)NC)cn2)ccc1F 86663,c1(C(N2C(C(=O)NCc3cocn3)CC(=C)C2)=O)c(O)ccc2ccccc12 86664,C1(CNC(C2C(Cl)(C(=O)OC)C2)=O)(NC(=O)C(O)P(C)(C)=O)CC2CCC1CC2 86665,C1(NC(Cc2cnc(C)s2)=O)COCCN(C(=O)C(c2ccc(F)cc2)(C)O)C1 86666,c1(N(C)C)ccccc1C(=O)NC1(CC(=O)NCc2ncsc2Br)CCC1 86667,c1(CC(=O)NCCN(C(C2CC2(C)Br)=O)CC)cn[nH]c1 86668,c1(CCC(=O)NCCN(C(C2(C)CCC(=O)C2)=O)CC)ccc2ccccc2c1 86669,C1(CNC(C=C(C)C(C)(C)C)=O)CC2CN(C(C3CC3C(=O)NCCO)=O)CC12 86670,c1(N2CCCC(CO)CC2)ncnc2ccc(O)cc12 86671,CN1CCc2[nH]nc(C(=O)Nc3ccc(CN=[N+]=[N-])nc3)c2C1 86672,c1(C(N2CCC(NC(C(C(C)C)SC)=O)C23CC3)=O)ccc2c(C)noc2c1 86673,CCC(CCC(=O)N(c1ccccc1)CC)NC(C1CCCS1)=O 86674,N(C1COc2ccc(Cl)cc21)C(C(Cc1ccccc1Br)NC(C)=O)=O 86675,c1(NC(C(=Cc2cocn2)C)=O)cnc(OC2CCOC2)c(C)c1 86676,c1(C(=O)NCC2(C)CN(C(c3ccc(F)nc3)=O)C2)cnc(O)c(Br)c1 86677,S(=O)(=O)(c1ccc(NCC2CSCCS2)c(C#N)c1)NCCCC=CC 86678,c1(OC)ccc(C)cc1C(=O)NC1CC12CC(NC(=O)Cc1csc(S)n1)C2 86679,C12(C(=O)NCC3C(NC(C=C(CC)CC)=O)CCCC3)CC3CC(CC(C3)O1)C2 86680,c1(C(N2CC3CCC2CC3)C(=O)NC(CC)C)ccc2cccc(Br)c2n1 86681,N1(C(c2c(NC)cncc2)=O)CCC(C(=O)NCCCS(C)=O)C12CC2 86682,Cc1ncnc(C(=O)NCc2ncoc2CCNC(=O)Cn2cc(Cl)cn2)c1C 86683,C(CCC(=O)N(C1CCCCC1)CCNC(=O)C=CC1(C)COC1)N(C(C)=O)C 86684,N1(n2cc(C=O)scncc2)CC(F)(F)CC1CNC(C1(C(F)F)CCCC1)=O 86685,C(=O)(CCC(=O)NCc1cn(CC(N2CCC(C)CC2)=O)nn1)NC.C1C(=O)N1 86686,c1(C(=O)NCC2N(C)CCN(C(CCSC)=O)C2)nc(C)c(C)nc1C 86687,C=C(Cl)CCC(=O)NC(C1CCCC1)CNC(=O)CNC(c1cccnc1)=O 86688,c1(NC(CN(C(=O)C(C)SC(F)(F)F)C(CC)C)=O)ccc(OC)c(OC)n1 86689,c1(C(=O)NC(C)CCN(C(=O)C(C)CC(F)(F)F)C)ccc2nnc(S)n2c1 86690,c1(C(=O)NC(CNC(c2cocn2)=O)C2CCC2)cc(Cl)nnc1O 86691,c1(CN(C)C(=O)NCC2CC2c2cn[nH]c2)cccc(O)n1 86692,c1(C(C)OCC)nc(C2=NOC3(CCOC3)C2)n(-c2nccn2C)n1 86693,c1(NC(C2(C(=O)OC)CC2)=O)cn(C)c(NC(c2cocn2)=O)n1 86694,CC1=C(C(=O)NCCOC2CCN(C(c3oc(C)nc3C)=O)C2)CC1 86695,N1(C(c2[nH]cc(C(C)=O)c2)=O)CC(C(=O)NC2CCOC(C)C2)CC1(C)C 86696,c1(N2CCCC(C(N)=O)C2)nc2ccc(Cl)cc2c(=NCCSC2CCCC2)[nH]1 86697,C1(CNC(C(CSC)(C)C)=O)CN(C(=O)C(C)(CO)NC(C)=O)CC1O 86698,c1(OC)cc(C(N2CCN(c3ccc(C(F)(F)F)nc3)CC2)=O)ccc1N 86699,c1(C(N(C)CC2CN(C(C3CCOC3)=O)C2)=O)csnc1Cl 86700,n1(CC)nnc2cc(C(N3CCCCCC(NC(C4CC(F)C4)=O)C3)=O)ccc12 86701,CCCCC(O)CC(=O)N1C2CCC1(CNC(=O)CN(c1ccncc1)C)CC2 86702,CC(CCCc1cn(CCc2ccn(C)n2)nn1)C(=O)N(CC#CC1CC1)CC 86703,C(=O)(C1=C(C)Oc2ccccc2C1)N1CCC(C(C)NC(CC(=O)OCC)=O)C1 86704,N1(C(C(C2N(C(C(CC(C)C)OC)=O)CCC2)(C)C)=O)CC2(CCNC(=O)O2)C1 86705,N1(C(CCCC#C)=O)CCCC(C2CCN(C(c3cscc3Cl)=O)C2)C1 86706,C1(C)(CC(=O)NCCC(=O)NC(c2ccn(C)n2)C)OCCO1 86707,N1(C(c2c(CC)occ2)=O)CCC(C(=O)NCC(=O)N(C)C)C12CCC2 86708,N1(C(C2CC2C2CC2)=O)CCC12CCN(Cc1cccc(F)c1O)CC2 86709,N1(C(c2c(CCC)n(C)nc2)=O)CCCN(C(=O)CC=C(Cl)Cl)CC1C(C)C 86710,c1(N(C)C)ccc(Cn2nc(-c3cccc(F)c3)nc2-c2cccnn2)cc1 86711,C1(C(=O)NC2(C3N(C(C=CC(C)=O)=O)CCC3)CC2)C(C=C(C)C)C1(C)C 86712,S(=O)(=O)(c1cc(Cl)c(Br)cc1F)N1CC(C(=O)Nc2cncnc2O)SCC1 86713,c1(C2C(C(=O)NCC(=O)N(C)Cc3ccccc3)C2)ncccc1Br 86714,c1(C(N2CCN(C(C(CC)C)=O)CC2CC(=O)NC)=O)ccnc2c1CC(=O)N2 86715,C(=O)(C(CC1CC1)NC(C1CCNC1=O)=O)NCC(c1cccs1)C 86716,c1(C(C(=O)O)NCc2cnc3cccnc3c2)cccc2ccccc12 86717,N1(C(C(C)(C)OC(C)=O)=O)CCC(C(F)F)(CNC(C2CCC3CCC23)=O)C1 86718,c1(NC(=O)NC)cccc(C(N2CC3CC3(CNC(=O)CN(C)CCO)C2)=O)c1 86719,c1(CC(=O)NCc2ccc(CNC(=O)CC3(O)CCC3)cc2)cc(Cl)cc(Cl)c1 86720,c1(-c2cn(CCN3C(N4C(=O)OCC4)COCC3)nn2)ccc(F)c(Br)c1 86721,N1(C(Cc2c(C)cco2)=O)CC2CC(C1)C2NC(=O)CNS(=O)(=O)N(C)C 86722,CC1(NC(=O)Cc2cnsc2)CCCCC1C(=O)NC1C=CCCC1CO 86723,C1(NC(CC(c2cccc(F)c2)C)=O)COc2ccc3ccccc3c2C1 86724,Cc1c(C(N2CC(C)N(C)C(C)C2)C(=O)NCCC2CC2)cc(F)cc1[N+](=O)[O-] 86725,CCCCCCC(C)CC(=O)NCC1(NC(c2cc(O)ccc2C)=O)CCOC1 86726,N12CCN(CC1)C(=O)C(C)N1CC2C1.c1(OC)ccc(C(F)(F)C(=O)OC)cc1 86727,n1(CCC)ccc(=NC(=O)C2CCC(C(C)C)N2C(C2CC2C#N)=O)[nH]1 86728,C1(CN2CCCC(n3cc(C4(S(N)(=O)=O)CC4)nn3)C2)COc2ccccc2O1 86729,c1(C(NNC(c2n(C)nc(S(C)(=O)=O)c2)=O)=O)cc(O)nc2ccccc12 86730,C(=O)(CC(O)C(C)CC)NCC(CC(=O)N(CC(C(=O)NC)C)C)O 86731,C(C(CNC(=O)CCNC(=O)OC)S(C)(=O)=O)NC(C=CC(CC)C)=O 86732,CCC(C(=O)NC1CN(C(C2(c3cccc(Cl)n3)CC2)=O)CC1O)C(C)(F)F 86733,C1(NCc2c(C)csc2Cl)CCN(C(=O)OCc2ccccc2)CCC1CO 86734,N1(C(C2CCC(F)(F)CO2)=O)CCC2(CC1)CCN(C(C1C=CCCC1)=O)C2 86735,c1(C(=O)NC2CC(NC(C3C(C(=C)C)OCC3)=O)C2)csc(=NC2CC2)[nH]1 86736,CS(=O)(=O)c1ccc(F)cc1C(=O)NC1CC(F)CN(C(C2CCC(=O)N2)=O)C1 86737,C1(CN(C)C(c2cnn(C3CCC3)c2)=O)CN(C(C2CC(F)C(=O)N2)=O)CCO1 86738,c1(NC)ccc(C(=O)NC(C(=O)NCc2cccc(Cl)n2)C(C)C)nc1 86739,CC1OC2(CNC(=O)C(C)NC(C)(C)C)CC1(NC(C1CCN(C)C1)=O)C2 86740,C1(NC(C(CCSC)O)=O)CCN(C(c2ccc(Cl)s2)=O)C12CC2 86741,C=CCC(C)(C(=O)NC1(CNC(=O)C(C)CC)CCC1)N(C)C 86742,C(=O)(C1Cc2ccc(C)cc21)N1CCC(NC(C(CC)CC)=O)(CF)C1 86743,c1(C(=O)NC2C(NC(c3c(C)noc3C3CC3)=O)CC2)onc2ccccc12 86744,C1(C(N(C)CCc2ncccn2)=O)CN(C(C2(C)CNC(=O)N2)=O)CCO1 86745,c1(C(N2CCC(NC(CC(=O)N(C)C)=O)CC2)=O)noc2c1CCCC2 86746,CC1(C)CCC(C(=O)NC2CCN(C(=O)CC3(C(F)(F)F)CNC(=O)C3)C2)O1 86747,S(=O)(=O)(C=Cc1ccccc1)NC1CC(NCC(=O)Oc2ccccc2)C1 86748,N1(C(c2cc(CNC(C(CC3CC3)OC)=O)[nH]n2)=O)CCC(C)(F)C1 86749,N1(C(c2ccnc(OC)n2)=O)CCN(C(c2nc3c(s2)COCC3)=O)C(C)C1C 86750,C1(CNC(C(CSC)(C)C)=O)CC(C)CN(C(=O)CC2CC(F)C2)C1 86751,C(CC(=O)NOCC(C)O)(C(F)(F)F)NC(C(C)NC(=O)OCC)=O 86752,C(=O)(C1=CCCC1(C)C)NC(C(C)C)CNC(c1cc(OCC(F)F)ccn1)=O 86753,C1(C(N2CCC(C(C)(C)C(=O)O)CC2)=O)(OC)CCCOC1 86754,C1(C(=O)NC2CC(C)CC2O)CC2(CCN2C(=O)OC(C)(C)C)CN1C(=O)C1CC1 86755,Cc1nnc(NC2CCCN(C(c3nc(C)n4ccccc34)=O)C2)c(C#N)c1C 86756,O(NC(=O)C(C)(C)CCCNC(=O)CCC(C)CC)C(C=C)C 86757,c1(NC(=O)NCc2nccc(OC)c2)ccc(I)cc1Br 86758,C1(C)(NC(C)=O)CN(C(C)=O)C1.C12(CC1)C(=O)OCC(=O)N2C.C(C)(C)(C)O 86759,C1(F)(C(=O)NC2CC(NC(c3cc(C(=O)OC)[nH]c3)=O)C2)CCS(=O)(=O)C1 86760,c1(OC)ccnc(C(=O)NCC(C)N(C(=O)CC(C)n2ccnc2CC)C)c1F 86761,C1(CC(=O)NC(C(=O)NCC(N2CCCCC2)C)CO)CCC(C)(C)C1 86762,Cc1ccc(CN2CCOCC(C(=O)NCC3=CCCCC3)C2)c(C)c1 86763,N1(C(C=CC)=O)CCOC(CN(C)NC(C2CC2C(N)=O)=O)C1 86764,C1(N(C)C(=O)C2CC2)CC12CCN(c1cc(=O)n(-c3ccccc3)[nH]1)CC2 86765,C1(NC(C2(CC=C)CCCC2)=O)CN(C(C2CC2=C)=O)CC(C)(C)C1 86766,N1(C(C2(COCC)CC2)=O)CCC(NC(=O)C(C(C)C)NC(N)=O)C1(C)C 86767,N1(C(c2n(CC)ncc2)=O)CC(NC(c2cc(Cl)no2)=O)CC12CCOCC2 86768,c1(C(C(=O)NCC2C(NC(CC(C)SC)=O)C2)N(C)C)c(F)cccc1F 86769,C1(NC(C=CCC)=O)CN(C(c2ccc(-n3ccnc3)cc2)=O)CCC1C 86770,C1(CNC(C=C(C)C)=O)(NC(C2CCCC(=O)N2)=O)CCCCC1C 86771,c1(CCNC(c2n(CCC)nc(C)c2)=O)c(Cl)cccc1Br 86772,c1(C(N(CC(C)NC(=O)Cn2cc(C#N)cn2)C)=O)ncccc1OC(F)F 86773,c1(SC)ccc(C)c(C(N2CCCC3(NC(c4ccns4)=O)CC23)=O)c1 86774,CS(=O)(=O)c1ccc(CN2CCC(O)(C(=O)Nc3ncc(I)nc3Cl)C2)cc1 86775,c1(C(N2CC(NC(c3c(C)ccc(C#N)c3)=O)C2)=O)ccc2c(=O)ccoc2c1 86776,C(C)(CCC(=O)NOCCCCC1CC1)NC(c1cc(CCC)[nH]n1)=O 86777,C1(NC(C2(CCC)CC2)=O)CC2CC1CC2C(=O)NC(CO)C1(C)CC1 86778,C1(CN(C)CC2CCN(C(c3ccccc3)=O)C2)CCS(=O)(=O)N1 86779,C1(NC(C2CCCCS2)=O)CCC2(CC1)CN(C(c1ccc(C3CC3)cn1)=O)C2 86780,C1(NC(c2cc(C=C)cc(F)c2)=O)CC(C2CCN(C(=O)CC3=CCCC3)C2)C1 86781,C=CCC(CNC(=O)Cc1ccn(C)c1)C(=O)N(c1ccc(C)cc1C)C 86782,C1(COC)CC(Cn2cc(C(C)OC)nn2)N(C(=O)CCC2CC(F)(F)C2)C1 86783,N1(C(CCC(=O)NCCC)=O)CCC2(CC2)CC1C(=O)NC1CC1CN(C)C 86784,c1(C(=O)NC(C2CC2(C)C)CC)c(CNC(=O)CCSC)cnn1C 86785,CS(=O)(=O)CCC(=O)N1CCN(C(=O)COC(F)F)C(C2CCC2)C1 86786,N1(C(c2ccc(C)cc2O)=O)CC2CCC(C1CO)N2C(=O)Cc1cccnc1 86787,C12(C(N(C(C)CCNC(=O)C(C)C3CCOC3)C)=O)CC=CC(C1)OC2 86788,Cc1ccc(C(N2CC(N(C)C(C3CCOCC3)=O)C(F)C2)=O)c(N)c1C 86789,C1(C(=O)NC(C(=O)NC)C)CC(F)(F)CN1Cc1cccc(I)c1O 86790,c1(NC(C(c2ccnn2CCSC)N(C(C#C)(C)C)C)=O)cccc(Cl)c1 86791,N1(C(C2C(C)C2C)=O)CCC(CCCNC(C2(C)CCCOC2)=O)CC1 86792,c1(C(N(CCNC(c2ccccc2)=O)CC)=O)ccc2nnn(C)c2c1 86793,C1(CNC(c2c(C)[nH]nc2Br)=O)COCCN(C(C2CCC(=O)N2C)=O)C1 86794,c1(OC)cc(C(=O)NCC2(C)CCCN2C(C2CC3(CC3)C2)=O)n(C)n1 86795,c1(C(N(C)Cc2cn(C(C)C)nc2)=O)cccc2c1CCO2 86796,C1(C(=O)NCCCOCCNC(C2C=CC=CC=C2)=O)CCC2(CCOC2)O1 86797,C(=O)(C(CCC(C)C)NC(C1CCC(=O)C1)=O)NC1(COC)CC1 86798,N1(C(C2C(C(N)=O)COC2)=O)CCC(C2CN(C(C3CCCCO3)=O)C2)CC1 86799,C1(NC(c2ccc(C(=O)OCC)[nH]2)=O)CCN(C(C2CC2OCC)=O)CC1 86800,C1(NC(C2(CC)CCCC2)=O)CCN(C(c2ccnn2CC(F)F)=O)CC1CO 86801,Cc1cnccc1C(=O)NCC1C2CN(C(c3cc[nH]c3)=O)CC12 86802,C1(C(=O)NC(CCC)C2CCC2)CCC(O)CN1C(C1CC2C=CC1O2)=O 86803,C(CCC(O)CO)N(C(CC1(C)N(C(C=CC=CCC)=O)CC1)=O)C(C)C 86804,N#Cc1cccc(F)c1NC(C1CC(F)CN1C(c1ccc(S)cc1)=O)=O 86805,C1(NC(C2(CNC(CCc3cc(C)on3)=O)CCC2)=O)CCCC1C1CC1 86806,N1(C(=O)OC(C)(C)C)CC(C(N2CCC3(CCC3O)C2)=O)C(C2CCCC2)C1 86807,C(=O)(C(CC(C)(C)C)OC)NC(C(=O)NCC(COC)(C)O)(C)CO 86808,C1(C(=O)NCCCN(C(=O)CC2CCCC(=O)N2)C)Cc2c[nH]cc2S1(=O)=O 86809,N1(C(CN2C(C)CC2)=O)CCC(CCNC(C2CC2C(=O)NCCN(C)C)=O)C1 86810,C1(C(=O)NCCCN(CCCNC(C2(C(C)C)CC2)=O)C)CCCC1(C)C 86811,C1(CNC(C=CS(C)=O)=O)CC(C)(C)CN1C(=O)Cc1nc(=N)[nH][nH]1 86812,C1(NC(c2c(N)c(Cl)ncc2)=O)CC12CCC(NC(C1CC1C(F)(F)F)=O)CC2 86813,c1(OC)cc(Br)c(F)cc1NC(=O)CC1CCCN1C(c1ccc(C)cc1I)=O 86814,CCS(=O)CC(=O)N1CCC(C(=O)NC(C)C(C)(C)C#N)(CF)C1 86815,N1(C(c2cnn(C)c2C#N)=O)CCCC2(CCCN2C(C2CCC2(C)C)=O)C1 86816,Cc1ccc(NC(=O)C(C)(C2CC2)N(C(=O)C(O)C(F)(F)F)C)cc1Cl 86817,c1(C(=O)NCC(CN(C)C(C2CC2(C)Br)=O)O)ccc(N)cn1 86818,C1(NC(C(C2CC2)OCC)=O)CC(C)(NC(C2CC(O)(CCC(C)(C)C)C2)=O)C1 86819,c1(CNCC2(C(=O)NC(C=C)CO)CC2)csc(Br)n1 86820,CN1N=C(CC(=O)N2CC(=O)NCC2C(N2CC3C(C(N)=O)C3C2)=O)CC1=O 86821,Cc1cc(F)c(C(=O)NCC2CC3CCC2N(C(c2csc(Cl)c2)=O)C3)c(F)c1 86822,C#CC1(CC)COCCN1C(=O)N(C1CCCN(C(c2ccccc2F)=O)C1)CC 86823,c1(N2CCC(C(C)(C)C)(CNC(C3(F)C(C)OCC3)=O)C2)nc(Cl)c(C#N)s1 86824,C12CCC(CC1)C(=O)NC2=O.N1(CC)CC=CC1Cn1cc(C2(F)COC2)nn1 86825,C(=O)(C(F)C(C)(F)F)N1CCC(CC(=O)N(C2CCS(=O)(=O)C2)C)CC1 86826,N1(C(C2(CC=C)CN(C(=O)CC3(O)CCOC3)C2)=O)CCC12CN(C)C2 86827,N1(C(C(C=C)OC)=O)CCC(C(=O)NC23CCCC2C3)C12CCC2 86828,Cc1cc(C(=O)NCC(C)(O)CNC(=O)CCSCC2CCCO2)nn1C(C)C 86829,C(=O)(CCC(C)(C)C)N(CCCCN(C(=O)CC(O)c1cnc(Cl)s1)C)C 86830,C1(C(NOCCCN(C)C)=O)CCOCCN1C(=O)CC1CC(=O)NC1=O 86831,N1(C(c2ncccc2F)=O)CCC2CC2(C(=O)NCC(Cl)Cl)CC1 86832,c1(OCCC(N2CCC(CC=C)(NC(=O)C(C)CSC)C2)=O)cc(F)ccc1F 86833,c1(CC(N2CC(N(C(C(CCC)C)=O)C)C(O)C2)=O)c[nH]c2ccc(OC)cc12 86834,c1(N(C)C)cnccc1C(=O)NC1CN(C(C2CCC23CCC3)=O)C1 86835,C(CC(C(=O)N(C1COC(C)(C)C1)C)NC(c1cc(C2CC2)[nH]n1)=O)=CC 86836,CC(C(=O)N1CCSCC1CCNC(c1csc([N+](=O)[O-])c1)=O)P(C)(C)=O 86837,C(C(C)(C)C(=O)NCC(C(=O)N(C)C(C1CCCC1)C)N(C)C)OC(C)C 86838,C(C(C)(C)CC(=O)Nc1cn(C)nc1C)NC(C1(CC)CCCCO1)=O 86839,c1(C(=O)NC2C(CNC(C(C)OCCCCCC)=O)CC2)ccn2cccc2c1 86840,C1(CNC(c2cnn(C)c2C(=O)O)=O)CCC2(CN(C(=O)OC(C)(C)C)C2)O1 86841,N1(C(C(C=CC)O)=O)CC2CCN(C(c3nn(C)c(Cl)c3Cl)=O)C2C1 86842,c1(C(N(C2CCC(NC(C3CC4(C3)CC4F)=O)CC2)C)=O)cc(N)c(Cl)c(O)c1 86843,c1(C(N2C(CN(C(c3cccc(C#C)c3)=O)C)CCC2)=O)ccc2c(c1)OCC2 86844,Cc1cnc(C(=O)NCC2(C(N3CC(C)(CO)C3)=O)CCC2)c(C)c1 86845,N1(C(C=C(CC)CC)=O)CCCC(O)(CNC(=O)CC2CCCN(C)C2)CC1 86846,N1(C(C2(C)CCN(c3nc(SC)c(F)cn3)C2)=O)CCC2(CCCO2)C1 86847,c1(CCC(=O)Nc2cc(OC)c(F)cc2)ccc2[nH]ccc2c1 86848,c1(C(=O)NC2CN(C(C(C=C)(F)F)=O)CC2C(F)F)ccc(Cl)c(C)c1N 86849,N1(C(C=C)=O)CCc2c(NC(C3(C)CCCOC3)=O)cccc21 86850,CC1CCC(C(=O)NC2(CO)CC(F)(F)C2)N(C(c2cn(C)cn2)=O)C1 86851,C1(CNC(C=CCOC)=O)CCCC12CCN(C(C1C3CCCOC13)=O)CC2 86852,Cc1cc(OCC(N2CC3CC2CC3NC(=O)CCC(C)(F)F)=O)ccc1Cl 86853,Cc1cc(C(=O)NC2CC3CC2CN3C(C2(C)CCC2)=O)c(F)cc1F 86854,N1(C(Cn2c(C)cnc2)=O)CC2CCC1CN2C(C1CCOC(=O)CC1)=O 86855,C(CCCCCN=c1[nH]nco1)N(C(c1nc(CCC)sc1)=O)C 86856,CC1CCn2c(C(=O)NC3CCN(c4cc(C5CC5)nc(Cl)n4)CC3)cnc2C1 86857,c1(OC)cc(C=CC(N2CCN(C(=O)C=CBr)C(CCO)C2)=O)ccc1O 86858,CCCC(C(=O)N1CCC12CN(C(=O)C(C)Cc1ccnn1C)C2)S(N)(=O)=O 86859,c1(C(N2C(C)CCC(CNC(CSCC(=O)OC)=O)C2)=O)cnn2ccccc12 86860,N1(C(c2c(C)ccc(Br)c2)=O)CCN(Cc2ccc(C3CC3)s2)CC1C#N 86861,c1(NC(C(c2cnc(CC)[nH]2)N2CCCC2C(=O)N(C)C)=O)ccc(F)cc1C 86862,C(=O)(C1(CC)CCCc2ccccc21)Nc1ccc(C(c2n(C)ccn2)O)cc1 86863,C1(C(=O)NCCC(C)SC)N(C(c2cc(C)cc(O)n2)=O)CCCC1(C)C 86864,C(=O)(C(CNC(c1ccc(COC)o1)=O)CC(C)C)NCCCCC(=O)NC 86865,c1(C(N2CC(OCCC(=O)NC3CC(C)(C)OC3)C2)=O)cc(F)ccc1Cl 86866,CN1CC2CN(C(C3OCCC3C(C34CCC(C3)C4)=O)=O)CC2(C)C1 86867,CCCC(C)(C)CC(=O)NC1(C2CN(C(c3nc[nH]c3C(F)(F)F)=O)C2)CC1 86868,C(CNC(=O)NC1CCCCC1n1cccn1)(CC)(CC)OCC 86869,C1(C(N(CC(C)N(C(C=COCC)=O)C)C)=O)CC(=O)N(C(C)(C)C)C1 86870,c1(C(C)=O)ccc(CN2CCC2CNC(=O)CCC2CC=CCC2)cc1C 86871,C1(NC(c2nc[nH]n2)=O)CCN(C(=O)C2CCCN2Cc2ccccc2)O1 86872,c1(C(=O)NCC(CN(C(c2cc(CC)sn2)=O)C)C)ccc(C)nc1 86873,c1(N2CC3CCCC(NC(Cn4c(C)nnn4)=O)C3C2)ncc([N+](=O)[O-])cc1C#N 86874,C1(n2cnnn2)(NC(=O)Nc2ccc(OC3COC3)cc2)CCCCC1 86875,C(=O)(C(C)(C)C(=O)NC)N(CC(CN(C(C(CC)n1ccnc1)=O)C)O)C 86876,C(C(C)C(=O)NC1CC(C(C)NC(C2CC2C(=O)OC)=O)C1)OC 86877,N1(C(c2ccc(=O)oc2)=O)CC2(C1)CN(C(c1ccc(Cl)c(Cl)n1)=O)C2 86878,C1(CC(=O)NC(CNC(C(COC)(C)OC)=O)(C)C)CCCS(=O)(=O)C1 86879,N1(CCOCC=C)C(=O)CN(Cc2cnn(C)n2)C1=O 86880,C1(C(=O)Nc2ccc(COC)cc2)C2CC1N(C(=O)Nc1cnn(C3CC3)c1)C2C 86881,c1(C(NCCC(C(C)CN)C(=O)O)=O)cc2n(n1)CCCN2 86882,c1(C(=O)NCC2OCCN(C(C(CC)=CCCC)=O)C2)ccc2c(c1)ncn2C 86883,C1(O)(CNC(C(C(C)(C)C)SC)=O)CC2CCC(C1)N2C(=O)Cc1cncn1C 86884,N1(C(c2c(C)ccc(F)c2)=O)CC2(CCN(C(=O)CC(C)C3CCCO3)CC2)C1 86885,C(=O)(CC(C(C)OC)NC(C1(CO)COC1)=O)NCCCOC 86886,Cc1ccc(C(C)C(N2CCN(Cc3nccs3)CC2)=O)cc1 86887,CC1CN(Cc2cc(C#N)ccc2OC(F)F)c2cccnc21 86888,C=CCC(CC(=O)N(C)CC1CC(O)C1)NC(C1CC2(C1)CC2(F)F)=O 86889,c1(C(=O)NC(C2CCOC2)CNC(CCOCC)=O)c(O)cc(Br)cc1F 86890,Cc1cc(F)c(C(=O)NC2CCCC2NC(=O)Cc2ccsn2)cc1F 86891,N1(C(Cc2cnc(C)[nH]2)=O)CCC(N(CCO)C(c2nccn2C)=O)CC1 86892,C1(C(=O)NCc2ccccn2)CSCCN1C(=O)CC1CC2C=CC1C2 86893,CC1(C)CCCC(C(=O)NC2CC3(C2)CC3NC(c2csc(C3CC3)n2)=O)CC1 86894,Cc1cc(Cl)c(C(=O)NC2C3CC2N(C(c2ocnc2C(F)(F)F)=O)C3)s1 86895,Cc1cccc(C(F)C(=O)NCCCCCNC(C2CS(=O)C2)=O)c1 86896,N1(C(C(C)(C)C2CCC2)=O)CC(CNC(=O)CCc2cc[nH]n2)C2(CCC2)C1 86897,c1(CC)noc(C(=O)NCC(C(C)C)NC(=O)CC2CCCOC2)n1 86898,N1(C(C2(C=C)CCC2)=O)CCCC(N(CCF)C(=O)Nc2cncc(C)n2)C1 86899,CC1(C)CC(C)(C(=O)NC2CCSCC2)CN1C(=O)CC1CC(F)(F)C1 86900,c1(C(=O)NCC(c2ccc(O)cc2)O)n[nH]c2c1CN(C(=O)Cc1ccco1)C2 86901,N1(C(Cc2n(C)ncc2Cl)=O)CCCC2CN(C(c3csc(O)n3)=O)CC12 86902,CS(=O)CCCCNC(C1C=CCN(C(=O)C=CCF)C1)=O 86903,N1(C(C(C)C2(O)CCC2)=O)CC2(CCC2)CC1C(=O)NC1C2CCCOC12 86904,N1(C(CCC2N(C(C(CSC)OC)=O)CCCC2)=O)CC(=O)NC(C)C1 86905,C1(CNC(C(c2ccc(Cl)cc2)CC)=O)C2CN(C(=O)CSC(C)C)CC12 86906,c1(CCC(=O)N(C2CC2)Cc2cccnc2S)ccc(S(=O)(=O)NC2CC2)cc1 86907,CC1CCN(C(c2ccccc2Cl)=O)CCN1C(=O)C1=CS(=O)CCC1 86908,C1(NC(C2ON=C(CC)C2)=O)CC2CC1CC2C(=O)NOCC(F)(F)F 86909,C1(OC)CCC2(C(=O)N(C3CN(C(=O)CCCc4sccc4C)C3)C)CC12 86910,Cc1cc(C)n2nc(C)c(C(N3CCC(C)(NC(=O)C(C)S(N)(=O)=O)C3)=O)c2n1 86911,c1(C(C)NC(c2c(O)ncc(C(C)C)c2)=O)ccc2ccccc2c1 86912,C(C(C)(COC)CC)NC(C1(C)CN(C(c2nc(COC)oc2)=O)C1)=O 86913,c1(NC(c2cn(CCO)nn2)=O)nc2ccccc2n1CCCCCC 86914,N1(C(C2OCCC(C)C2)=O)CCC2(CCC2CNC(=O)CN2CCCCC2)CC1 86915,Cc1cc(F)cc2c1CCC2NCc1nc(Br)cs1 86916,N1(C(CCC(C)(C)C)=O)CC(NC(=O)CN=c2cc[nH]cc2)CC2(CCC2)C1 86917,N1(C(CN2CCN(C(C3CCCN(CC)C3)=O)CC2)=O)CC2C(C1)C2(C)C 86918,C(=O)(C1=Cc2ccccc2C1)NCC(CC(=O)N(CC(F)F)C)C1CCC1 86919,C1(CCNC(=O)Cc2csnn2)COCCN1C(=O)CC1(CC2CC2)CCC1 86920,c1(C(=O)NC2C(NC(COCc3cccc(OC)c3)=O)C2)cc(N)cnc1Cl 86921,CCCC(C(=O)NCC1(COC)CN(C(=O)C#CC2CCCO2)C1)C(C)C 86922,C(CC1CCC1)(C(=O)NCC1CCCC1)NC(C(C)OCCCC)=O 86923,c1(C(=O)NC2CC(F)(CNC(C3CCC(C)C3)=O)C2)ccc2n[nH]cc2c1 86924,N1(C(C=CC(C)(C)SC)=O)CCCCC1CC(=O)NCC(c1ncc[nH]1)C 86925,CC#CC1CCN(C(=O)C(F)CC2CN(C(c3cnn(CC)c3)=O)C2)CC1 86926,C1(C(N2C3(CN(C(=O)CCN4CCCCCC4)C3)CC2)=O)CC2CCCCN2C1 86927,N1(C(CN(C2CCCC2)C)=O)CC2C(CNC(C3CCC(C)(C)C3)=O)C2C1 86928,C1(NC(C2CC(Cl)(Cl)C2)=O)CCC2(CCCN(C(c3ccncc3)=O)C2)C1 86929,c1(NC(C(CCSC)NC(=O)Cc2sccc2C)=O)cc(C)cnc1C 86930,N(C1c2ccccc2CC1NC(=O)C(C)C(O)CC)C(c1cn(CCC)nc1)=O 86931,C1(C(=O)NCCCOC)CCC=CC1NCc1ccc(C)cc1 86932,c1(C(N2CCCC(NC(C3C4COCC34)=O)C2)=O)ccc(C(F)(F)F)cc1Br 86933,N1(C(CC(C)C)C(=O)Nc2ccc(Cl)cc2F)CCS(=O)(=O)CC(C)C1 86934,N1(C(C(CC2(OC)CCC2)N)=O)CCN(C2CC2)C(C)C1 86935,CC(O)CCCC(=O)N(C(C)CCNC(C1(S(C)(=O)=O)CCC1)=O)C 86936,C1(C(N(CC(C(=O)Nc2c(CCC)cccc2)C)C)=O)CC(=O)OC1(C)C 86937,c1(C(=O)NCC(CNC(CN(C(=O)OCC)C)=O)(C)F)ncncc1C 86938,C(=O)(C(CO)C(C)(C)C)N1CCCC(F)(CNC(c2c(SC)scc2)=O)C1 86939,C(=O)(C1=NOC(C)(C)C1)NC1CN(Cc2nc(C)on2)C(C)CC1 86940,CC(CC(F)F)C(=O)N1CCCCC(N(C(=O)COCC2CC2)C)C1 86941,CC(C)S(=O)(=O)CC(=O)NC(C)C(CO)NC(c1ccccc1Br)=O 86942,c1(SCC(=O)NCC2C(NC(c3n(CCOC)ncc3)=O)C2)ccc(F)cc1 86943,c1(CC)ccccc1CC(=O)NC(CN(C(=O)C(CC)NC(C)=O)CC)CC 86944,C1(N(C)CC)CCN(C(C2CCOCC2NC(=O)CC2CCN(C)C2=O)=O)CC1 86945,Cc1ccncc1CN1CCC(NC(=O)NCC2CCCO2)C1 86946,CS(=O)(=O)C1CCCC1C(=O)NCC1(NC(C2CC3(CSC3)C2)=O)CCOCC1 86947,C1(C(=O)NCC2CN(C(c3c(SC)ccs3)=O)CC2O)CC2(CCC2)CCO1 86948,c1(C(=O)NCCCC(c2ccccc2)NC(CN(CC)CC)=O)sc(C)cc1Cl 86949,C1(C(=O)NC(CCSC)C(N)=O)CC12CCN(C(c1ccccc1Cl)=O)CC2 86950,C1(C(=O)NCCCOCCN(C(CC=C=C)=O)C)Cc2ccccc2O1 86951,CC(C)C(C(=O)N1CCC(c2cccc(F)c2)(NC(c2cocn2)=O)C1)NC=O 86952,C(=O)(N=c1[nH][nH]c2c1CN(S(=O)(=O)CCCCCl)C2)c1cc(C)c(C)nc1 86953,C12(CC)CN(C(=O)CCCSC)C(CNC(c3sc(C)c(C)c3C)=O)(C1)C2 86954,C1(C)(C(=O)NC(CC)CSC)CC(NC(=O)COC2(C)CCC2)C1 86955,c1(Nc2cccc(CC(N)=O)c2)ccc([N+](=O)[O-])c(OC2CNC2)c1 86956,c1(C(=O)NC2CC(C)(CNC(C3(C)ON=C(C)C3)=O)C2)cc(C)c(C)cn1 86957,N(C(=NCCN1CCSCC1)NC1CCS(=O)(=O)C1)C1(C)CC1.N1(C)CCOCC1 86958,c1(COC)cc(C(=O)NC(CC(=O)NC2CC(C(F)(F)F)C2)C2CC2)no1 86959,N1(C(C2(OC)CCSC2)=O)CC2CCC(C1)C(NC(=O)C1=COCCC1)C2 86960,C1(c2cn(CC(=O)OC)nn2)CCCCC1OCC(=O)NCCN1CCCOCC1 86961,N1(C(c2c(C)[nH]c(C#N)c2)=O)CCN(C(=O)C(C)(C)C2CCC2)CCC1C 86962,N1(C(Cn2cc(CNC(C3(CC)CCCC3O)=O)nn2)=O)CCC(C)C(C)(C)C1 86963,N1(C(C(C=C)(C)C)=O)CCC(C)N(C(c2ccc(C(F)(F)F)s2)=O)CC1 86964,c1(C(=O)NC2CC(C)(NC(c3c(NC)cnnc3)=O)C2)cc2c([nH]1)CCCC2 86965,N1(C(CCN(CC)CC)=O)CC=CC1CNC(c1ccsc1C(F)(F)F)=O 86966,C(=O)(C1=CCCC1)NCCC(C)NC(C1CC1c1cccs1)=O 86967,c1(NC(=O)NCc2ncc(OC)cc2C)ccc2ccccc2c1 86968,CC1CCC(NC(=O)CCN2CCN(C)CC2)CN1C(C1SCCS1)=O 86969,c1(NC(c2ccc(ONC3CC(F)C(C(=O)O)C3)cc2)=O)ccccc1OC(F)F 86970,C(CC(O)C(=O)NC1COCCC1C(=O)NC(CO)CCO)N(C)C 86971,c1(CNC(c2c(C)n[nH]c2)=O)cc(F)cc(F)c1.c12c[nH]nc1C1CCN(C1)C2=O 86972,N1(C(c2nc(C(C)(F)F)sc2)C(=O)NCCCC2CC2)CCC2(C=CCO2)CC1 86973,C(C)(C(C(=O)NCCC(C)N(C(=O)CSc1cn[nH]c1)C)N(C)C)OC 86974,c1(C(C)C(=O)NCC2CCCC2n2cccn2)ccc2c(c1)CCC2 86975,c1(C(=O)NCC(C)(C)OCCNC(C2CCN(C)C2)=O)cccc(C#N)c1 86976,N1(C(CS(C)(=O)=O)=O)CC2CCN(C(=O)Cc3ccc(O)c(O)c3)CC2C1 86977,CC1=NNC(=O)C1CCC(=O)NCC(C1CCC1)NC(C1(n2cccn2)CC1)=O 86978,N1(C(C(CN(C)C)NC(C2ON=C(C)C2)=O)=O)CC(S(C)=O)C1 86979,C1(C(=O)NC(C2CN(C(=O)C(=C3CCCCC3)F)CCO2)C)(CC)CCOCC1 86980,C1(C(=O)Nc2c(C(=O)OC)scn2)CCN(C(c2cc(F)nc(F)c2)=O)CC1O 86981,N1(C(C2(C3CCCO3)CC2)=O)CCC(F)(CNC(C2(CC#N)COC2)=O)CC1 86982,N1(C(CC(C)=C(C)C)=O)CCN(C(c2cnn(C)c2)=O)CC(O)C1 86983,C1(C(=O)NCCNC(=O)CCOC2CN(C(c3ccoc3)=O)C2)OCCCO1 86984,C(=O)(CCCCCCCO)NC1CN(C(=O)NCc2cn(C(C)(C)C)nc2)C1 86985,C1(NC(=O)C=Cc2ccncc2)CN(C(=O)Cc2csc(S)n2)C2(CCOC2)C1 86986,C(=O)(C1=COCCO1)N(CCN(C(=O)C(N1C(C)CCC1C)C)C(C)C)C 86987,c1(C(N2CCN(C(CN(C(CC=CC)=O)C)=O)CC2)=O)ccc2nc(O)[nH]c2n1 86988,C1(OCC)(NC(=O)NCC2COC3CC2C3)CCCCC1 86989,N1(C(C(CCC)OC)=O)CC(CNC(=O)CCn2cncn2)C2(CCOCC2)C1 86990,N1(C(CCN(C)CC)=O)CC2(CC(NC(=O)C(C)C3CC3)c3nccn32)C1 86991,C(=O)(CC(C1CCCC1)NC(=O)CC(C)c1cnn(C)c1)OC 86992,CON(C)C(=O)C1(NC(=O)C(O)C2CCCC2)CCC1 86993,c1(OC)cncc(C(=O)NCC(C(C)C)NC(C2CC2c2ccc(F)cc2)=O)n1 86994,C(=O)(C1Cc2ccc(Cl)cc21)N1C(C)(CNC(=O)CC2CC3(CC3)CO2)CCC1 86995,C1(Cc2cn(CCOCC)nn2)COCCN1C(c1cc(-c2ccco2)[nH]n1)=O 86996,C1(C(c2ccncc2)OC(=O)C2CC2)CCCN(C(C2(c3ccncc3)CC2)=O)C1 86997,N1(C(c2cccc(C(C)(F)F)c2)C(=O)NCCCC)CCCC(O)(C(N)=O)C1 86998,Cc1cc(=NCc2ccc(C(C)(C)C)o2)[nH]cc1S(=O)(=O)NC(c1ccco1)C 86999,c1(C(N=c2cc(C)o[nH]2)=O)cn2c(n1)CCCC2C(=O)O 87000,c1(NC(C2(C)CN(C(c3cc(F)c(F)cc3I)=O)C2)=O)ncc(Cl)cc1[N+](=O)[O-] 87001,c1(CC)sc(C(=O)NCC2CCN2C(=O)CC(C)F)cc1Br 87002,c1(N(C)Cc2c(OC)nsc2)nc(=NC2CCC(CN(C)C)C2)[nH]c2c1CCC2 87003,Cc1nc(C(N2CCC(F)(CNC(=O)CC3NC(=O)NC3=O)C2)=O)sc1C 87004,c1(C(=O)NC(C2CCCC2)CNC(C(C)c2ccsc2)=O)c(F)cccc1F 87005,C1(C)(C(N2CC(SC)C(N(C)C)C2)=O)COC(C)CO1 87006,c1(SC)nccc(N2CC(CNC(=O)C(c3cccc(F)c3)C)CC2C)n1 87007,C#CC1(N(C)C)CN(C(C2C=CCCN2C(C2CCCC2O)=O)=O)C1 87008,Cc1cc(CC(N2CC(C(C)(C)O)(CNC(C3(C)CC3(F)Cl)=O)C2)=O)c(C)s1 87009,CC1CC(CCNC(=O)Nc2ccnn2CC2CCC2)CCO1 87010,Cn1nccc1C1CC1C(=O)NC(C)(CNC(=O)COc1cccnc1)CO 87011,C(CN=C(NCC(F)(F)CO)N1CCN(Cc2ccc(Cl)cc2)CC1)OCC=C 87012,Cn1cc(CN2CCCC(NC(C3CNC(=O)C3)=O)CC2)c2ccc(F)cc12 87013,Cc1cc(CNC2C3CN(C(=O)C(c4ccccc4)N(C)C)CC23)c(C)s1 87014,N1(C(CC(=C)C)=O)CC(NC(C23CCC2CC3)=O)C(c2nccn2C)C1 87015,C(=O)(CCC(C)(C)C)NCCN(C(=O)Cn1cc(C2CCOC2)cn1)CCOC 87016,c1(C(C)C)ccc(C(=O)NCC2CCN2C(=O)CC2CCCCC23CC3)cc1F 87017,C(=O)(C(O)C(C(C)C)OC)N1C(C(=O)NCC(=O)NC)CC1 87018,Cc1ccc(F)c(-c2cn(CC3C=CCN3C(C3(C)CCC(C)C3)=O)nn2)n1 87019,c1(N(C)Cc2ccc(C)s2)nc(=NC2CC(C3CCCC3)C2)[nH]c2c1COC2 87020,C1(NC(c2noc(CC)c2C)=O)CCCC12CN(C(c1cnn(C3CC3)c1)=O)C2 87021,C1(NC(CNC(=O)OCC)=O)CC2CC(NC(C3(O)CCCCC3)=O)CC12 87022,C(=O)(C1=COCCO1)N(C1CCCN(C(c2nc[nH]c2C(C)(C)C)=O)C1)CC 87023,c1(OC)cc(CN2C(C(=O)Nc3ncc(F)cc3Cl)CC3CC23)cc(O)c1O 87024,C1(CNC(C(CC)(C)O)=O)CC(F)CN(C(=O)CCc2cncc(Br)c2)C1 87025,C(=O)(CC(C)C(C)C(C)C)NCC(CCOC)NC(c1[nH]c(C)cc1C)=O 87026,C1(OCC)CN(C(c2ccn(CC)c2C)=O)CC1CNC(=O)CC(C)(C)O 87027,c1(OC)cnc(C(=O)NCCCNC(c2cc(-c3cccs3)on2)=O)nc1 87028,C12(CNC(C3N(CC)C(=O)CC3)=O)CN(C(C3CCCO3)=O)CC(F)(C1)C2 87029,CC(C)C(O)C(=O)NCCC(C)N(C(=O)CC1(c2ccccc2)CS(=O)(=O)C1)C 87030,C(=O)(C(F)CC(C)(C)C)N(CC(=O)NCC1(C)CC1(C)C)CCOC 87031,CC1(CNC(c2cnn(CCF)c2)=O)CCCN(C(C23CCC(CC2)CO3)=O)C1 87032,c1(C(N2CC(NC(Cc3c(COC)cccc3)=O)C2)=O)cc(Br)cnc1N 87033,C1(NC(CC2(C=C)CC2)=O)CN(C(c2cc(CC)ccn2)=O)CC1C 87034,N1(C(Cc2cc(C)sc2C)=O)CCC(C)C(NC(=O)Cc2cc(O)nc(O)n2)C1 87035,C1(C(=O)NC(C2CCCN2C(=O)CCc2ccc(O)cc2)C)OCCN(C)C1=O 87036,O=C1CC(=O)NC(C(=O)NC(CNC(c2ncnc(O)c2F)=O)C2CCC2)C1 87037,CCC(CC(=O)NCC1(CNC(=O)C(C)(C)c2cccs2)CC1(F)F)SC 87038,CN1C(=O)C(N(C(=O)CNC(=O)C(C)(C)C)C)CCc2ccccc21 87039,N1(C(C(C=C)OC)=O)CC2CC1CN(C(=O)C(C)NC(C)(C)CC)C2 87040,C1(NC(CS(=O)(=O)NC)=O)CC2CC(NC(c3ccn(CCOC)n3)=O)CC12 87041,C(N=C(NC1CCC1)N1CCC(NC(N)=O)C1)c1ncc(CC)s1 87042,C(=O)(C(F)CCC(C)C)NC1CN(C(c2c[nH]c(=NC)o2)=O)C(C)C1 87043,c1(C(N2CCC3(CC2)CC3CO)C(=O)NCC(C)C)nccc2cc(Cl)ccc12 87044,C=CCC(C)(CC)C(=O)N1CCCN(Cc2cn(-c3ccccn3)nn2)CC1.OCC 87045,O=C1COc2c(Nc3cc(NCC4CC5C(C4)C5(F)F)ncn3)cccc2N1 87046,C(=O)(C(Cn1cccn1)NC(=O)C(c1ccccc1)=O)N(C)C 87047,N1(C(CC(C)OCC)=O)CCN(C(c2ccc(OC(C)C)nc2)=O)CC12CC2 87048,C1(C(N2CC(O)(C(C(=O)N(C(C)C(=O)NC)CC)F)C2)=O)CC12CCOCC2 87049,C1(NC(c2cccc(C(C)=O)c2)=O)CCN(C(=O)CN(C)C2CC2)CC1C 87050,CC(CCC(C)(C)C)C(=O)NCC1CC(C(N2CC3(CC(F)C3)C2)=O)C1 87051,C1(N(C(c2c(C)n(C)nc2)=O)C)CCCC2CN(C(c3cnc[nH]c3=N)=O)CC12 87052,c1(CS(=O)(=O)NC2(COC)CC(O)C2)cccc(C(F)F)c1 87053,Cc1sc(C(=O)NC(C)CCCNC(=O)C(C(C)O)N(C)C)nc1O 87054,C1(COC)(NC(c2cc(C)nn2C)=O)CCN(C(C2CC23CCC3)=O)CC1 87055,c1(C(N(CCNC(=O)C(=O)NCC(F)F)CC2CCCC2)=O)cc([N+](=O)[O-])n[nH]1 87056,C=CCC(C(=O)NC1CC1NC(=O)Cc1sccc1C)NC(=O)OC(C)(C)C 87057,C1(NC(C2CC(CNC(C(n3ccc(C)n3)C)=O)OC2)=O)CCC=CCCC1 87058,CC(CC(F)F)C(=O)N1CC(NC(c2cnc(Cl)s2)=O)C(C(F)F)C1 87059,C1(C(N(CCN(C(C(CCC)CC)=O)CC)CC)=O)CCC2(CCCCC2)CC1 87060,c1(C(N2CCC(COC)(NC(=O)CC34CC(C3)C4)CC2)=O)cc2c([nH]1)CCCC2 87061,c1(-n2c(C3(Nc4c(C)noc4)CCC4CC34)nnn2)ccc2c(c1)OCO2 87062,CC1CN(C(C2(CNC(=O)C(C3(O)CCCC3)F)CCCCC2)=O)CC1O 87063,Cc1cc(C)c(C=CC(=O)NC2CN(C(c3cc(C)[nH]c3C)=O)C2)c(C)c1 87064,O=C(CC1=CCN(C(C2CCCC2O)=O)CC1)Nc1cccn2nccc12 87065,C1(NC(c2ccc(CCC)o2)=O)CN(C(c2ccc(NC)cn2)=O)CC1C1CC1 87066,C12(C(N3CC(F)(CNC(c4cc(CC)ncc4)=O)C3)=O)CCC(CC1)OC2 87067,C1(C(C#C)C)CCN(C(C2CCC2CNC(C2(C)SCCCS2)=O)=O)CC1 87068,C1(C(=O)NC(CC(C)NC(c2cc(C)n(C)c2)=O)C)CN2CCN1CC2C 87069,CON(CCC(=O)Nc1cnc2ccnn2c1)C(=O)CC1CC2C=CC1C2 87070,c1(C(C(N2C(C(C)NC(=O)Cc3cn(C)nn3)CC2)=O)C)noc2ccccc12 87071,N1(C(C(C=C=C)C)=O)CC(C2CCN(C(=O)Cn3ccc(=O)n(C)c3=O)CC2)C1 87072,C#Cc1ccc(NC(C23CC(C)(CN2C(=O)C(C)(C)CCCOC)C3)=O)c(C)c1 87073,C1(C2CCN(C(C3CCC(C)O3)=O)C2)CN(C(=O)CCc2ccn(C)n2)CCO1 87074,C12(NC(CCC(=O)NC)=O)CCC(CN(C(=O)CC3CCCC3)C1)C2 87075,C(=O)(CCCC(=O)NC(CNC(=O)CSCc1cccs1)C(C)C)NCCC 87076,CS(=O)(=O)c1ccccc1N1CCN(C2C3CC(O)C2NC3)CC1 87077,N1(C(=O)NCc2nocc2C(=O)NCc2ncoc2CC2CC2)C(=O)CCC1=O 87078,Cc1nnc2n1CC(C(N1CC3(C1)CN(C(=O)CC(C)C)CC3CO)=O)N(C)C2 87079,c1(C(=O)NOCC(F)(F)F)ccc(C2SC(=O)CS2)cc1 87080,C1(CNC(=O)NC(c2ccc(F)cc2)C2CC2)CCC2COCC2O1 87081,C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CCCC=C)C(=O)N1CCOC(C)C1C 87082,c1(C(N2C(CCNC(CCC(=C)C)=O)CC(OC)C2)=O)ccc(S(N)(=O)=O)s1 87083,c1(C(=O)NCC2N(C(C(C)=C3CCC3)=O)CC(C)CC2)ccc2sccc2c1 87084,c1(C(=O)NC(C2CCCN2C(=O)Cc2cncs2)C)nc[nH]c2ncnc1-2 87085,C(=O)(C1CCc2nccn21)NC1(C)CCCN(C(c2cccc3ncsc23)=O)C1 87086,CON(C(=O)C1=CCC(NC(C23CCC(C2)C3)=O)C1)C1CCC1 87087,c1(CN2CC(NC(C(CCC)C)=O)C(F)C2)cc(Br)cc(Cl)c1O 87088,N1(C(C(C2CCCOC2)OC)=O)CCC(N2CCN(C(C)=O)CC2)CC1 87089,c1(C(=O)NCC2(CSC)CC2)ccc2n[nH]cc2c1.C1(C(=O)N)(CF)CCC1 87090,N1(CC)CCC(N=c2[nH]c3c(c(=NCC=CBr)[nH]2)COCC3)C(C)C1 87091,N1(C(Cc2cc(C)on2)=O)CC(NC(C2(C)CC2(F)F)=O)C(C)C1 87092,n1(CC)ccc(C(=O)NCC(O)CNC(c2scc(C)c2Cl)=O)cc1=O 87093,CN1CCOCC1CC(N1CCC(O)(CNC2(c3cccnc3Cl)CC2)C1)=O 87094,Cc1nsc(NC(C2(CNC(c3nn(C)c(C)c3Br)=O)CC2)=O)c1C#N 87095,N1(C(C=C(C)Cl)=O)CCCC2(C1)CN(C(c1cnc3c(Cl)cccn13)=O)CCO2 87096,C=CC1(C(=O)NCC2C3CCCCCC23)CCN(C(=O)CC2CCC(C)(C)O2)C1 87097,c1(C(=O)NCC(=C)CCNC(c2cc(-c3cccnc3)on2)=O)oc(C)cc1C 87098,C1(C(=O)NCCCCC(=O)NC)CCC2(CC2)N1C(C12CCCC1OCC2)=O 87099,C1(CN(C(=O)CC2CCCCC2O)C)COCCN1C(=O)CC1CC=CC1 87100,Cc1nn(C)c(C)c1C(=O)NCCCN(CCCNC(c1ccsc1)=O)C 87101,c1(C(N2CCC(CC#C)(C(=O)N(CCF)CCOC)C2)=O)cc(F)ccc1F 87102,N1(C(c2cn(C3CC3)cn2)C(=O)NC(CC)C)CCOC(c2ccnn2C)C1 87103,C=C1COc2c(-c3nc(CCCN)no3)cnn2C1 87104,C1(NC(CCCC#CC)=O)C2CCN(C(c3c[nH]ccc3=O)=O)CCC12 87105,n1(CC)c(C(N2CC(=O)CC2C(=O)N(C)CCF)=O)cnc1O 87106,C1(C2CCN(C(C(CC)C)=O)C2)CCCCN1C(=O)CSCCN(CC)CC 87107,c1(C(=O)NCCn2cc(CNC(CC(C)OC)=O)nn2)cccnc1S 87108,C1(F)(CNC(c2cn[nH]c2)=O)CN(C(=O)C(F)(F)c2c[nH]nc2O)C1 87109,c1(COC)cnc(C(=O)NC(C2CCN(C(=O)CCF)C2)(C)C)s1 87110,N1(C(C(CNC(C2CCCC(F)C2)=O)N(C)C)=O)CCn2cncc2C1 87111,c1(C(=O)OC)ccc(OC(=O)N(C2COC(C)(C)C2)C)c(OC(F)F)c1 87112,c1(CC)ccc(C(N2CC(NC(C3CSCCS3)=O)C(F)C2)=O)cc1 87113,c1(C(C(N2CCC(CNC(C(CC)(C)C)=O)C2)=O)(C)C)ccc2ccccc2c1 87114,N12CCN(C)C(C1)C2=O.C1(NC(C2C(C)CC2)=O)COCC1F 87115,C1(C(N2CC(CC(C)NC(=O)COCCCN(C)C)C2)=O)CCC12CCOCC2 87116,C=CC1CN(C(=O)C(C(C)C)NS(C)(=O)=O)CC1NC(C1CC(=C(F)F)C1)=O 87117,n1(CCC(=O)OCC)nnnc1C(CCc1cnccn1)NCC(C)C(C)C 87118,C(=O)(C#CC1CCCOC1)N1CCC(C)C(NC(C2CC(F)(CO)C2)=O)C1 87119,C1(C(N(CC(F)F)C(C)C)=O)CCC(C)(C)N(C(=O)CC2CCCO2)C1 87120,c1(CNC(C2C(NC(c3cc(C)c(C)o3)=O)CCOC2)=O)nn(C)c(=O)n1C 87121,N1(C(c2cc(C)c(C)o2)=O)CC(O)CC1(C)C(=O)NCCCCF 87122,c1(CCC(=O)NC(C)CC(C)NC(c2cncc(F)n2)=O)ccc(C#N)cc1 87123,O=C(C1c2ccccc2CN1c1ncnc2c1CCC2)N1CCC2(CCC2)C1 87124,N1(C(C(C2CC2)NC(c2ccc(C3(C)CC3)cc2)=O)=O)CC(O)CC12CCC2 87125,c1(CC)cc(C(=O)NC2COCCN(C(C3C(C)(C)C3(F)F)=O)C2)c(C)nn1 87126,C1(C(N2CC(C#C)(F)C2)=O)CC2C=CC1N(C(=O)CC1C(C)(C)C1(C)C)C2 87127,O=C(CCS(=O)(=O)c1ccc(F)cc1)NC1CCN(C(C2CC2(F)F)=O)C1 87128,c1(CNC(c2cnn(C)c2)CC)cccc(CC(F)(F)F)c1 87129,C(=O)(C(c1cn[nH]c1)N(Cc1cccs1)CC1CC1)NCC(=C)C 87130,c1(C(N(CC)CC2CCCO2)=O)oc(CNC(=O)CC(C)C2CC2)nc1C 87131,C1(NC(COCCCC#C)=O)CCCC(C(N2CCC(C)(C)C2)=O)CC1 87132,N1(C(c2cnc(CC)nc2)=O)CCCC(C)(C)C1C(=O)NCC(F)CO 87133,c1(N2C(C(NOC(c3ccccc3)C)=O)CC(O)C2)ncnc2cc(C)nn12 87134,c1(C(N2CCCCC2)=O)cc(C)c(Cl)c(C)c1.C(C(=O)OC(C)(C)C)N(CC)CC 87135,C1(CNC(C(CC)NC(c2n[nH]cc2Cl)=O)=O)C2CCCCCC12 87136,N1(C(C(C)=C(C)C)=O)CCC2(C1)CN(C(=O)Cc1ccc3nn[nH]c3c1)CCO2 87137,N1(C(COCC=C)=O)CCC(CCNC(c2cc(C)nnc2O)=O)C(F)(F)CC1 87138,c1(C(=O)NC2C(NC(C=C(C)Cl)=O)CCC2)[nH]c2ccc(Cl)cc2c1Cl 87139,C1(F)(C(=O)NC2CC(NC(CN(C)C3CC3)=O)C2)CC1(Cl)Cl 87140,CC1(C)c2ccccc2CC1C(N1CC2CCC(C1)N2C(C1(CF)CC1)=O)=O 87141,c1(C(=O)NC(CCOC)CNC(C2CCCS2)=O)cncc2nc(C)[nH]c12 87142,C(C)(C)(C(c1ccc(CS(C)(=O)=O)s1)N(C=O)Cc1cnc(C)o1)OC 87143,C(C(=O)NCC(CO)NC(=O)COCc1cccc(C)c1)(C(C)(C)C)NC(C)=O 87144,c1(C(=O)NC2C(OC)CN(C(c3csc(CC(C)C)n3)=O)C2)cnc(C)c(C)c1 87145,CP(C)(=O)c1cnn(CC(N2CCCC(C(=O)Cn3cncn3)C2)=O)c1 87146,N1(C(CNC(CC)=O)=O)CC(CNC(c2cnccc2Cl)=O)C2(CCC2)C1 87147,C1(C(N(CC(=C)C)CCOC)=O)CCCC(NC(c2ccncc2)=O)C1 87148,c1(CN2CCCC(C(=O)Nc3cc(F)ccc3I)C2)ccc(F)cc1[N+](=O)[O-] 87149,N1(C(c2c(C)nccc2)=O)CCC2C1CCN2C(c1cc2cccnn2n1)=O 87150,c1(OC)cc(F)c(C)cc1NCc1ccnc(Br)c1Br 87151,C(CCCC(=O)N1CCC(F)(CNC(c2cc(C(C)(C)C)no2)=O)C1)OCC 87152,N1(C(C2(C#N)C(C)C2)=O)CC2CCC1CN2C(c1nc(C2CC2)cs1)=O 87153,O=C1CCC(O)CN1CC1COCCO1.c12cn(nn1)CCC(=O)NC1CC2C1 87154,C(C(CC(F)(F)F)NC(c1snc(O)c1Cl)=O)NC(C(C(C)C)OC)=O 87155,C1(O)(C(C)NC(CCOCCC)=O)CCN(C(=O)CNC(=O)C(F)(F)F)C1 87156,CCC(C(=O)NC1(CNC(=O)Cc2ncoc2C)CCCC1)NC(C)=O 87157,C1(NC(CC2(C#N)CC2)=O)CC(O)CN(C(=O)Cc2csc(C3CC3)n2)C1 87158,N1(C(CCCCOCCC=C)=O)CCC2CN(C(=O)CC(COC)COC)C2C1 87159,C(=O)(C(CCS(C)=O)N(C)C)NC1CCC1CF.c12ccccc1CN(C)C2=O 87160,C1(NC(CC2(C)CCN(C(c3cc(CCO)on3)=O)C2)=O)(CO)CC2CCCC12 87161,C1(CNC(C=CCOC)=O)CCCC2CN(C(C3(C)CC3(F)F)=O)CC12 87162,CC(C)CC(O)C(=O)NCC1(F)CCCN(C(c2nnc(S)n2C)=O)C1 87163,Cc1ccc(O)cc1C(=O)N(CCC(=O)NC1CCCCC1(C)O)CC1CC1 87164,CCC(C(=O)N(C1CCCCN(C(c2cc(C)nc(O)c2)=O)C1)C)C(C)(F)F 87165,N1(C(CNc2cncc(C(N)=O)c2)=O)CCC(NC(c2ccoc2Cl)=O)C12CC2 87166,N1(C(C2CCC(C(=O)OC)O2)=O)CC2(CNC(=O)C(O)C(C)(C)C)CCC1CC2 87167,N1(C(C(Br)=C(C)C)=O)CC2CCC(NC(=O)Cc3cccc(F)c3F)CC2C1 87168,c1(C(=O)NC(C2CCCCN2C(=O)Cc2ccccc2)C)cc2c[nH]cnc-2n1 87169,c1(C(CNC(C=CC)=O)NC(=O)C=C2CCN(C)CC2)cc(F)cc(Br)c1 87170,C(=O)(C1CCCc2nccn21)N1CCC(CNC(c2ccc(CC)cc2)=O)CC1 87171,N1(C(CC=CC)=O)CCC2CCC12CNC(c1c(O)cccc1Cl)=O 87172,C(CCCC(=O)NCC(C)(Cn1cccn1)NC(=O)CCc1ncco1)SC 87173,C(=O)(C(C(=O)NC1(C(=O)NC2C=CCCCC2)CCCCC1)OC)OCC 87174,c1(C(=O)NCCC(=C)CNC(=O)CCOCCC(C)C)cn(C)nc1O 87175,C=CC(C)(CC)C(=O)NCc1csc(CNC(c2[nH]c(C3CC3)nc2C)=O)n1 87176,N1(C(C)C)CC(C(=O)N(C2CC(NC(C34CC(CCO3)C4)=O)C2)C)CCC1=O 87177,C1(NC(CC2N(C)CCC2)=O)CCC2(CC1)CN(C(=O)CC1CC3(CCC3)C1)C2 87178,C1(C(=O)NC2CCCN(C(CCn3ccc(C)n3)=O)C2)CN2CCC1(C)CC2 87179,Cc1oc(C#N)cc1C(=O)NC12CC1CN(C(c1ccnn1C1CCCC1)=O)C2 87180,C(=O)(C(C(C)C)NC(N)=O)N(CCCN(C(C(C)=CC)=O)C)C 87181,c1(C(N2C(COC)(CNC(c3n[nH]cc3OC)=O)CCC2)=O)cc(C)ncc1C 87182,N1(C(CCC(CCC)CC)=O)CCC2CCCC(C1)N2C(=O)CC(O)CC(C)C 87183,C(CCC(=O)NC(c1cn(C)nn1)C(=O)NCc1ccn(CC)n1)=CCC=C 87184,N1(C(CCCOCC)=O)CCN(C(c2ccc(C)cn2)=O)C2CC12 87185,N1(C(c2cc(OC)ns2)=O)CCSCC1C(=O)NC(c1nnc(O)o1)C 87186,C1(C(N(C)CC2CN(C(=O)C(O)c3ccsc3)C2)=O)CCCN1C1CCCCC1 87187,[N-]=[N+]=NC1CCN(C(=O)COCCNC(C2(F)CC=CCC2)=O)C1 87188,c1(C(=O)OC2C=C(Br)C2)cc2cc(Cl)ccc2[nH]1 87189,N1(C(C2C(C)CC2)=O)CCN(CC(=O)N(C)C(c2cnnn2C)C)CC1 87190,N1(C(C2(CC(C)C)CC2)=O)CCC(NC(=O)C=Cc2ccc(Cl)s2)C(CO)C1 87191,c1(N(c2ccnc(C)n2)C2CC2)ccc(C(N2CCC(NC(C)=O)CC2)=O)nc1 87192,CC(C(=O)NCC1CC(NC(=O)Cc2cccs2)CCO1)C(F)(F)F 87193,C(=O)(C(C)S(C)(=O)=O)N(C(C)C(N1CCCC(CN=[N+]=[N-])C1)=O)C1CC1 87194,C#CCC(CC(=O)N(C1CC(NC(=O)CO)C1)C)NC(=O)CCSC 87195,C1(CC(N2CCC(NC(C3(F)CCOC3)=O)C(CO)C2)=O)CN2CCN1CC2 87196,c1(C(N2CCN(C(C3CC(C#C)(O)C3)=O)CC2)=O)cc(Cl)c(Cl)n1C 87197,c1(OC)c(C(N2CC3CCN(c4nccc(SC)n4)C3C2)=O)cccc1[N+](=O)[O-] 87198,c1(C(=O)NCC(CN(C(=O)CC23COC(C)(C2)C3)C)O)c(N)cccc1Cl 87199,C1(CC)C(C(=O)N(C(C)CN(C(=O)C=Cc2ccco2)C)C)CCN1C 87200,CC1=NNC(=O)C1CNC(c1ccccc1)Cc1ccc(F)cc1 87201,N1(C(C2=NNC(=O)C2)=O)CC2(CCC2)CC1CNC(C1CCOCC1)=O 87202,C(C(=O)NNC(=O)C#CC1(C)CCCO1)OCc1cccc(OC)c1 87203,Cc1noc(C(=O)N(C)CC2CCCCN2C(=O)COC2CCOC2)c1C 87204,C1(C(N2C(CNC(C3(OCC)CCSCC3)=O)CCCC2)=O)CCN(C)S1(=O)=O 87205,c1(C(=O)OC)cnc(NC(C2CCCC(NC(c3ccc(C)cn3)=O)C2)=O)nc1 87206,C#CC1(C(=O)NCCCCC2CCCC2)CCN(C(=O)C(F)C2CCOC2)CC1 87207,Cc1n[nH]c2cc(C(=O)NC(CNC(=O)CCC3CCCO3)C(C)C)ncc12 87208,C(=O)(C(=O)N(C)C)N(CC(C)N(C(C1C(CC(C)C)C1)=O)C)C 87209,c1(CN(CC=C)C)ccc(OC)cc1.c1(N2CCC2=O)ccon1 87210,N1(C(c2ncoc2C(F)(F)F)=O)C2CCCC1CC(NC(C1(O)CCCC1)=O)C2 87211,C(C)(C)(CCC(=O)NC1CC(C)CCC1O)NC(c1ncn(CC)c1)=O 87212,C1(C(C)C)CN(C(=O)C2=NNC(=O)C2)CCCN1C(c1ccc(Cl)c(CO)c1)=O 87213,Cc1ccc2c(C(=O)NC(CNC(c3cc(C)ccn3)=O)C(C)(C)C)c[nH]c2c1 87214,c1(C(N(CC(C)N(C(C(CC)OCC)=O)C)C)=O)ccc(-n2ccnc2)nc1 87215,C#CC(CNC(=O)C(C(C)(C)C)n1cc(C2(O)COC2)nn1)CC(C)(C)C 87216,S(=O)(=O)(c1ccc(C)cc1)C(N(CCC(=O)OC(=O)C(F)(F)C(C)O)C(C)=O)=O 87217,n1(CC(=O)NC2CC(NC(CCCn3c(C)ncc3)=O)C2)ncc2ncccc12 87218,N1(C(C2CC(=O)C2)=O)CCN(CC2CCCN(C(C3CC(F)(F)C3)=O)C2)CC1 87219,CC(C(=O)N1CC(CO)CO1)n1cc(C2(O)CCCC2)nn1 87220,c1(C(N(C(C)CNC(C2CCCCS2)=O)CC)=O)cccn2cc(C)nc12 87221,c1(CNC(C2=C(C)CCCC2)=O)n[nH]c2c1CN(C(c1csc(C)n1)=O)CC2 87222,N1(C(CC(C)(C)CC(F)F)=O)CCC2(CCC(CN=c3ccnc[nH]3)O2)CC1 87223,N1(C(c2c(SC)csc2)=O)CCC2(C1)CN(C(c1cc3occc3s1)=O)C2 87224,CCC(COC)C(=O)NCCC(C)N(C)C(C1CC=CCC1)=O 87225,C1(O)(C(C)NC(=O)C=CC(=O)N(C)C)CCN(C(C2CC(=O)CO2)=O)CC1 87226,O(C1CCc2c(Br)cccc21)C(c1ccc(C2CCCOC2)cc1)=O 87227,C1(NC(C2CCN(C(N)=O)C2)=O)CC2(CCN1C(=O)COC1CCCOC1)CC2 87228,C(c1c(F)ccc(Cl)c1F)=CC(N1CCC(NC(C(C)=C(C)C)=O)C1C1CC1)=O 87229,c1(C(N2C(C(=O)Nc3ccno3)CC3CC32)=O)ccc2nccc(Cl)c2c1 87230,N1(C(C=Cc2ncc(C)[nH]2)=O)CCOC(C)C1C(=O)NCCC(CO)C(C)C 87231,CCC(CCC(=O)NCC1(C(=O)NCCc2cc(C)ns2)CCC1)OC 87232,C(=O)(C#CC1CCCCO1)N1CCCC(CNC(c2c(C)cn(C)c2)=O)CC1 87233,Cc1nccc(CN(C)CC2CCCCN2C(c2ncoc2C(C)(C)C)=O)n1 87234,C1(NC(C=C(C)C)=O)CC12CCN(C(c1ccc(Cl)c(C)c1)=O)CC2 87235,c1(C(=O)NCCN(C(=O)CCc2cnoc2)CC(C)O)cccc2ccccc12 87236,Cc1cc(N2CCOC(CN(C)C(C3CC3Cc3ccccc3)=O)C2)nc(Cl)n1 87237,Cc1cnccc1C=CC(N1CCOC(CNC(c2nnc(O)cc2O)=O)C1)=O 87238,C12(C(=O)NC(C3CCCO3)CC)CCC(NC(=O)CCc3cn(C)cn3)(CC1)C2 87239,N1(C(C2=C(C)OCC2)=O)CCCC2CCN(C(c3c(C(F)F)cnn3C)=O)CC12 87240,C(=O)(C(COC)CC(C)C)NCC(CC)N(C)C(c1sccc1Cl)=O 87241,CC(CC(C)(F)F)C(=O)OCC1OCCCO1 87242,N1(C(CCc2cc(C)no2)=O)CC2CCC(C1)N2C(c1cc(C)c(Cl)cc1C)=O 87243,N1(C(CC(C)=C(C)C)=O)CCC2(CC2C(=O)Nc2ccc(O)c(Cl)c2)C1 87244,C12(C(=O)NCCn3c(C)nnc3)CCC(CC1NC(C1CC3(C1)CC(O)C3)=O)C2 87245,c1(C(N2C(CNC(=O)C3=COCCC3)CC(C)(C)C2)=O)ccc2c(c1F)CCC2 87246,C(=O)(CCCCN(C)C(c1ncccc1Cl)=O)NCC(CC1CC1)OC 87247,C(C(=O)N(CCC(=O)NCCCn1ccnc1)CCO)(C(C)C)NC(C)=O 87248,c1(C(=O)NC(CNC(C2CC(=C)C2)=O)(C)C2CC2)cc(CC)nnc1C 87249,c1(CNC(C2CC2)NC2C(NC(C3(C(N)=O)CC3)=O)CC2)c[nH]nc1C(=O)CO 87250,C#Cc1ccc(C(=O)OCC(C2CC3C=CC2C3)=O)cc1 87251,CS(C)(=O)=Nc1ccc(C(N2CCN(C(=O)CC3CCCC3)C(CF)C2)=O)cc1 87252,Cc1nc(C(=O)NC(CC(=O)N2CCC(n3cncn3)C2)C2CC2)c(C)o1 87253,c1(NC(C2CN(Cc3ncc(Br)cc3Br)C2)=O)ncnc2occc12 87254,c1(CC)ncncc1C(=O)NC(C1CCN(C(=O)CCc2cccnc2)C1)C 87255,C(C(C)C(F)C(=O)Nc1cn(C)nc1C#N)NC(c1ccnc(OC)n1)=O 87256,c1(COC)ccnc(NC(C2CCCC(NC(c3cscc3C)=O)C2)=O)c1 87257,C12(C(N3C(C)(C(=O)NC)CC3)=O)C(NC(=O)C(C)C#N)C3CC1C2C3 87258,C1(NC(C2(C)CC=CCC2)=O)CN(C(c2cc(Cl)cnn2)=O)CCC1F 87259,C1(NC(C(C)N(C)C)=O)CCN(CC2CCC(C)C2)CC1(C)C 87260,c1(C(=O)OCC)ccccc1N.c1cncc(OCC(=O)N(C2CC2)CC)c1 87261,Cn1nccc(C(=O)NC2CN(C(=O)Cn3nccn3)CC2O)c1=O 87262,N1(C(CC=C)=O)CC(NC(c2ccnc(CC(C)C)n2)=O)CC(F)C1 87263,N1(C(CCc2c(C)ncs2)=O)C2CCCC1CN(C(=O)CC1CCC3CC13)C2 87264,c1(CNC(c2ccc(Oc3ccc(OCC)cc3)cc2)=O)cncc(O)c1Cl 87265,C1(C)(C(=O)NCC(=C)CCNC(c2cc[nH]c2C(=O)OC)=O)CC(O)CN1C 87266,C1(CC(=O)NCCCN(CCC)C(C2CC2(C)C)=O)(OC)CCC1 87267,C12(OC)CCC(C(=O)NC3CCN(C(=O)CC4(C)CC4(Cl)Cl)C(C)C3)(CC1)C2 87268,N1(C(C2N(CCCC)CCCC2)=O)CCC(C)(C)C(C(=O)N(C)C)C1 87269,C(C(C(=O)N(C)CC1(O)CCOC1)C(C)(C)C)NC(C(C(=O)OCC)(C)C)=O 87270,c1(CC2(C(=O)NC(CC(C)NC(=O)CC3CCCC3)C)CC2)ccc(O)cc1 87271,c1(CC)cccc(C(=O)NC2CC(NC(=O)Cc3c(Cl)cnn3C)C2)c1F 87272,[N-]=[N+]=NC1CN(C(=O)NCCc2cnco2)C1 87273,N1(C(CCSCC)=O)CCN(C(c2cccc(C(F)(F)F)n2)=O)C(C)C1 87274,CC1(C)CCCC(CC(N2CCN(C(c3ccnc(S)c3)=O)CC2C2CC2)=O)O1 87275,c1(C(N2C(CNC(C(C)CC(F)(F)F)=O)CCCC2)=O)c2c(nn1C)CCCC2 87276,C(=O)(CC(C)C)NC1(C(=O)N(CC)CC)CSC1.C12(CC1)C(=O)N2 87277,c1(CC)nc(O)c(C(N2CCC3(NC(=O)CC4CCSCC4)CC3C2)=O)cc1C 87278,N1(C(c2ccc(C#C)o2)=O)CCCCC2C1CCCN2C(=O)C(F)C(C)C 87279,C1(NC(CN(C)C)=O)CC2(CCCN(C(=O)C3CC3)C2)C1 87280,Cc1scc(C(=O)NCC2CN(C(C3(Cl)CC3(F)F)=O)CC2O)c1N 87281,C(=O)(C(CNC(=O)CN1CCCCC1C)(CC)CC)NC(C#C)C(C)(C)C 87282,C1(CCC(=O)NC(C)(C)C)CCCCN(C(=O)CSc2nc[nH]n2)C1 87283,Cc1nc(N)c(CC(=O)NCC2C3CCC(C3)N2C(C2CC(F)(F)C2)=O)c(O)n1 87284,C1(NC(c2cnn(C)c2F)=O)CN(C(C2CC3CCC2O3)=O)CC2(CCC2)C1 87285,c1(C(C)C)cc(N2CCC(NC(=O)C3=CCCCC3)C(C)C2)n2ncnc2n1 87286,CC(C)CCCC(C)C(=O)N1CC(CNC(C2CCCCCCC2)=O)C(C)(C)C1 87287,C=C=C(C)CC(=O)N1CCC(N(C(=O)CCSc2ccccc2F)C)C1 87288,C1(CN(C(C(C)OCCC(C)C)=O)C)CN(C(=O)CC=CC(C)(C)C)CCO1 87289,CC1CCN(C(=O)C(=O)NCc2cc(C(F)(F)F)ccn2)CCS1=O 87290,c1(C(C(=O)N(CC(C)NC(c2c(C)ccnc2)=O)C)(F)F)cccc(F)c1F 87291,c1(C(N2CCC(C(=O)Nc3c(C)cc(O)cc3)C2)=O)c(F)c(F)c(O)c(F)c1F 87292,C1(NC(CN2C(C)CCC2)=O)CCC2(CC1)CC2NC(C1C2CC3C(C2=O)C13)=O 87293,c1(OC)ccc(C(=O)NCC#CC(=O)NCC(=O)NC2CCCC2)s1 87294,N1(C(C(=O)NCC)=O)CCOCC(C)(CNC(=O)CC2CCCCCCC2)C1 87295,c1(C(=O)NCC2CCC(F)(CNC(=O)CC34CCCC3C4)C2)ccc(F)cc1Cl 87296,c1(N(C(=O)C(=O)NCC(C2CC2)C2CC2)CC=C)c(CO)cc(Br)cc1C 87297,N1(CC)CC(NC(=O)C=CC2CCC2)CC1=O.c1(C2(N)C(OC)C2)ncc(C)o1 87298,N1(CC)CCCCC1C(N1CCCCC1C(=O)NC1CCC(OC)C1)=O 87299,C(CN=c1[nH]c(=NCCC2CCCCO2)[nH]c2cc[nH]c12)c1ccc(SC)cc1 87300,c1(-c2cn(C3CCC(C(=O)Sc4cccc(Br)n4)C3)nn2)cc(F)c(Cl)c(Cl)c1 87301,N1(C(CONC(=O)C2(CCC)CC2)=O)CCCC[Si](C)(C)C1 87302,CCCCN=c1[nH]c(=NCc2n[nH]c3c2COCC3)[nH]c2c1SCC2 87303,c1(C(=O)NCC2CCCCN2C(c2n[nH]cc2F)=O)c[nH]cc(Br)c1=O 87304,N1(C(CC(C(F)F)NC(c2cc(C)c(F)cc2)=O)=O)CCC2CCCC2CC1 87305,Nc1sc2c(c1C(N1CCC3(C1)CN(C(=O)C1=C(Cl)CCOC1)C3)=O)CCC2 87306,[N-]=[N+]=NCCCCCC(=O)N1CCOC(C2CN(C(=O)C3=NOCC3)C2)C1 87307,c1(C(=O)NCC2C3N(C(C4C(CCC)C4)=O)C(CC3)C2)ccc2oc(O)nc2c1 87308,c1(CC=C)ccccc1C(N1CCC(CNC(=O)C(C)n2cccn2)(OC)C1)=O 87309,C1(NC(=O)C=CC(F)(F)F)CCCCC12CCN(C(=O)C=Cc1cccs1)C2 87310,c1(OCCC)ccc(C(N2CCCC2CNC(=O)CC2CCOC2C)=O)cc1 87311,C(=O)(CCC=CBr)NC(C(C)NC(c1ccc(NC(=O)C2CC2)s1)=O)C 87312,Cc1nc(C(=O)NC(C)CN2CCN(C(=O)COC3CCCC3)CC2)c(C)s1 87313,N1(C(c2cc(C)c(Cl)s2)=O)CC2CC1CN2C(C1CC(C2CC2)=NO1)=O 87314,N1(C(C2CNC(=O)N2)=O)CC(C2CC2)(C(=O)NC2C3C=CC(C3)C2CO)C1 87315,c1(CC(=O)N(C(C)CCNC(C2CCCCO2)=O)C)c(F)ccc(Br)c1F 87316,c1(C(N(CCCCNC(C2CCC2)=O)C)=O)csc(C2CC2)c1 87317,N1(C(c2ccc(NC)cn2)=O)CCCC(CC(=O)NCC2(C)CC(O)C2)CC1 87318,C(C1=CCN(C(=O)C(O)CN2CCOCC2)CC1)NC(c1c(COC)cc[nH]1)=O 87319,c1(C(=O)NC2C(NC(c3sc(C(=O)OC)c(N)c3)=O)CC2)cn(C)c(=O)nc1O 87320,C1(C2CCOCC2)(CNC(C2(C)CCCCC2)=O)CCN(C(C2CC=CC2)=O)C1 87321,N1(C(C2N(C(CCC)=O)CCCC2)=O)CC2(CCCCN(C(=O)C(C)CO)C2)C1 87322,C1(=CC(N2C(c3ccc(OC)cc3)SCC2)=O)CC2CCC(N2)C1F 87323,C(=O)(CC(O)CC(C)(C)C)NCC(=C)CCNC(=O)Cc1cccnc1Cl 87324,C1(CNC(C(C)c2cn[nH]c2)=O)CC(O)CN1C(=O)CCc1cc(Cl)no1 87325,N1(C(C2CCC(=O)C2)=O)CCC2(CCCN2C(c2cscc2F)=O)C1 87326,C(=O)(CCCCCOC)N1CC(CC)C(C(N2CC(F)C(F)C2)=O)C1 87327,c1(NC(CCC)CCCNC(C2CCC2(C)C)=O)c([N+](=O)[O-])c(CC)nn1C 87328,CC1(CC(N2CC(O)(CCNC(=O)C(N)=O)C2)=O)CC1(F)F 87329,N1(C(CN(C)S(N)(=O)=O)=O)CCC2(CC1)CC2NC(=O)CCSc1nccn1C 87330,N1(CC(CC(=O)OC)NC(C)=O)CCCN(Cc2noc(C3CC3)n2)CC1 87331,C1(CNC(CN(C)C(c2ccccc2)=O)=O)CCCCC1NC(=O)CC(F)F 87332,c1(OC)ccc(C2(C(=O)NCCC(C)NC(=O)CC3CCC(=O)N3C)CC2)cn1 87333,CC(C)(CCC(=O)NC1(CNC(=O)C(O)(C2CC2)C2CC2)CC1)[N+](=O)[O-] 87334,CC(CC(=O)NC1CCN(C(C2CC2(F)F)=O)CC1C)C(F)F 87335,c1(C(C(=O)N2CC(F)C2)NC(CCOC(C)C)=O)cnn(C)c1 87336,C12(NC(c3c[nH]c(=O)cn3)=O)CCC1CN(C(=O)COCc1ccccn1)C2 87337,c1(C(=O)NC2CC(NC(CCCN(C(C)=O)C)=O)CC2O)cc2occc2n1C 87338,N1(C(c2cn(C3COCC3OC)nn2)C(=O)NCCCC)CCCC(OC)C1 87339,C(CN=c1cc(C)nc(C)[nH]1)C1(O)CCN(C(C=CC=CC=CC)=O)CC1 87340,C1(C(=O)NOCC2(F)CCC2)C2CCCC2CN1C(=O)Cc1ccccc1F 87341,CC1c2ccc(F)cc2CCN1CC(=O)N(c1cccc([N+](=O)[O-])c1)c1cncs1 87342,c1(C(=O)OC)c(OC)ncnc1Cl.c12cc(ncn1)NCCN2.C1(CN)CCOCC1 87343,CC(CC(C)NC(C1CCCN1c1cnccn1)=O)NC(=O)C(C)(C)C 87344,c1(C(=O)OC)nn(C)cc1NC(C1CCCN1C(=O)C=CC(C)(C)SC)=O 87345,c1(C(=O)NCCC(=O)NCCC)c[nH]nc1CNC(C)=O 87346,C1(C(=O)NC(c2ccccc2)CC)CC2(CCC2)CN1C(=O)C(CO)C(F)(F)F 87347,C1(C(=O)NCC2(F)CN(C(C(N3CCCCC3)C)=O)C2)CCC(=O)NC1 87348,C1(C2CCCN(C(=O)C(C)(C)CC#N)C2)(NC(C(c2ccncc2)C)=O)CC1 87349,CC1CN(C(=O)Nc2cccc(-c3ccc4c(c3)OCCN4)c2)c2cnccc2O1 87350,C(=O)(C(CNC(C1CNC(=O)N1)=O)CC1CC1)N(CC(C1CCC1)OC)C 87351,c1(C(=O)NCC2N(C(c3c[nH]c(=NC)s3)=O)CCCC2)cc(C)c(Cl)c(C)c1 87352,CC(CNC(c1ccc(O)cn1)=O)C(F)C(=O)NCCc1cccnc1F 87353,N1(Cc2c(OC)nccc2)CC2CC1CN2C(c1ccc(O)c(F)c1)=O 87354,c1(COC)nc(OC)cc(NC2CC(O)(CNC(=O)Cc3c(C)noc3C)C2)n1 87355,c1(C(C)NC(C(CC)NC(c2ccccc2)=O)=O)cc2ccccc2s1 87356,C1(C(N2CCN(C(CCOC)=O)CC2C)=O)CC2CC1C1C2C1(F)F 87357,C1(CC(=O)NCCC2(O)CN(C(COCC=C)=O)C2)CCOC(C)(C)C1 87358,C1(N(CC=C)C(=O)NC)CN(C(=O)C(CC)=CC)CCC1(C)C 87359,c1(C(N2C(C(C)NC(c3cc(Cl)cnn3)=O)CCC2)=O)cncc2nc[nH]c12 87360,CN1CC2(CN(C(=O)NCc3ccccc3N3CCOCC3)C2)OC1=O 87361,C1(c2nnnn2-c2ccccc2)(NCC(CC)(C)CO)CCS(=O)CC1 87362,CON(CCCO)C(=O)C1(CO)CCCN(C(c2cnnc(C)c2)=O)C1 87363,C1(CNC(C2CC(=C3CC3)C2)=O)CCCN1C(C1(c2cccnc2)CCCC1)=O 87364,CC1CN(C(c2cccc(O)c2)=O)CC1(C)C(=O)NC1CCC(C)(C)CC1 87365,c1(NC(C2(C)CCN2Cc2ccc(O)c(O)c2)=O)ccc(OC(F)(F)F)cc1Br 87366,C=C(C)C1CCC(C)CC1NCCCOc1ccc(Br)cc1 87367,c1(CC)oc(C(=O)NC2(C(=O)NCCCN3CCC(O)C3)CCN(C)C2)cc1C 87368,C1(CC)CCN(C(C)=O)C1C(=O)OCc1ccccc1.C1CS(=O)(=O)N1 87369,c1(CNC(C(C)Cn2ccnc2)=O)ncccc1C(=O)O 87370,c1(C(=O)NC23CN(C(C(CC=C)C)=O)C(CC2)CC3)cc(C#N)c(O)nc1N 87371,C1(N(CC#C)C(=O)OCC)CCN(C(=O)C(C)Cc2ccccc2)CC1 87372,N1(C(CC=CC=C)=O)CC2CC1CC2NC(C1(Cn2cccn2)CCCC1)=O 87373,C1(CN(C)C(c2scc(Cl)c2Cl)=O)CN(C(=O)Cc2cncs2)CCO1 87374,N1(C(C2CC(CC)(CC)C2)=O)CC(C(=O)NC2CCCC2O)CCC1C 87375,C1(C)(OC)CCCN(C(=O)CC=CCNC(=O)C2=C(C)OCC2)CC1 87376,Cc1c(C(=O)NCC2COCCN2C(=O)Cn2cc(Br)cn2)cncc1Br 87377,C1(CC)CN(C(c2cocc2C)=O)CCC1NC(C1(C)CC=CC1)=O 87378,c1(C(N2CCC(F)(CNC(C(CC)OCC)=O)C2)=O)cccc(S(N)(=O)=O)c1 87379,C(=O)(CCCCN(C(=O)C(C)(F)c1ccon1)C)NC(c1cc[nH]n1)C 87380,c1(OC)ccc(CCC(=O)NC2CN(C(C3CCSC3)=O)C2)cn1 87381,CC(CC(=O)N(C)CC1(O)CCN(C(=O)C(F)(F)CO)C1)C(F)(F)C(F)(F)F 87382,c1(C(N)=O)ccc(C=CC(=O)NCC2CC(NC(c3cscc3Cl)=O)C2)o1 87383,N1(CC2(NC(C=COCC)=O)CC2)CCN(C(=O)C(F)(F)c2ccccn2)CC1 87384,Cc1cc(C(=O)NCC(=C2CN(C(=O)Cc3ccn(C(C)C)n3)C2)F)n(C)n1 87385,C(CO)(CCCCNC(C1(C)COC(=O)OC1)=O)NC(C=COCC)=O 87386,C1(CNC(CC=CC=C)=O)(CNC(=O)CCNC(=O)CC(C)C)CC12CCC2 87387,CC(C)CCCCC(=O)NC1CC1CNC(c1ccnc(OC(C)C)c1)=O 87388,CC1(C)CC(C)(C(=O)NCCCC2CN(C(c3cc(=O)cc[nH]3)=O)CCO2)C1 87389,Cc1cc(C(N2CCCC2CNC(c2ccc(=N)[nH]c2)=O)=O)ccc1Br 87390,c1(C(=O)NCCOC2CN(C(=O)CCOC3CCC3)C2)nnc2ccccc2n1 87391,C12(C(=O)NCCCCNC(Cc3cc(C(C)C)no3)=O)CCCC1CC2 87392,c1(C(N(CCCc2cccc(C)c2)C)=O)c2c(nn1C)CCCC2 87393,CCCC(C)C(CC)(c1nnnn1CCOCC1CC1)NCc1ccc(=N)[nH]c1 87394,N1(C(c2nc(Cl)sc2Cl)C(=O)NC(CC)(C)C)CCC2(CCCC2)CC1 87395,c1(CNC(CN(C(=O)CNC(=O)NC)CCC)=O)ccc(C)nc1 87396,c1(C(C)NC(=O)Cc2cccc(C(F)(F)F)n2)ccc(S(C)(=O)=O)c(OCCN)c1 87397,CS(=O)(=O)CC(=O)NC1CCCCC1NC(=O)CNC(=O)C(F)(F)F 87398,C12(CNC(c3n(C)cnc3)=O)COCCN1CCN(C(c1cnsc1)=O)C2 87399,CCC(CC(C)C)C(=O)N(CC(C)(C)CNC(=O)CC1CCC(C)(C)CC1)C 87400,c1(CC)ccoc1C(=O)NCC1(CNC(C2CN(C3CCC3)C2)=O)CCC1 87401,N1(C(c2cc(C3(C)CC3)on2)=O)CCCC(C2CC2NC(=O)CCP(C)(C)=O)C1 87402,C1(NC(C2CCC(=O)S2)=O)CCc2nncn2C1 87403,C(=O)(C(C)(F)C(=O)NCC(C)(C)NC(c1ccnc(O)c1)=O)OC 87404,N1(CC(C)(O)C2CCCC2)CCCC(c2n[nH]c(=N)o2)C1 87405,c1(C(=O)NC(C2CCN(Cc3cccnc3Br)CC2)C)cc(Cl)cnc1Br 87406,C1(NC(C(CC)NC=O)=O)C=CCN(C(=O)COc2cccc(OC)c2)C1 87407,N1(C(CCCC=C)=O)CC(C2CC2)(C(=O)NC2CCCOC2)C1 87408,Cc1ccc2c(c1)C(C(=O)NC(C)(C)CNC(C1CC1c1ccccc1)=O)C2 87409,c12ncccc1CN1CCC(C1)N2.C1(N(C)CC)CCN(C)CC1 87410,C(=O)(NNc1ncc(Br)c2ccccc12)C(C)(C)CNC(=O)OC(C)(C)C 87411,C1(CCC(N2CC(CC(C)NC(=O)CN(c3ccccc3)C)C2)=O)CCCN1C 87412,C12(C(=O)NCC(C)(C3CC3)NC(=O)CC34COCC(C3)C4)CCC(CC1O)C2 87413,N#CCCCC(=O)NC1CCN(C(=O)COc2ccc(Cl)cc2)C1 87414,c1(CC(N2CC(CNC(C3(C)CC(C#N)C3)=O)C2)=O)ncn2c1CCCC2 87415,c1(CN2CC(NC(=O)C3CC3)C2)nnn(C)c1C(=O)NC(c1cc(CC)[nH]n1)=O 87416,C=CC1(C(=O)NCCC(C)CCO)CCN(C(=O)CCOCCOC)C1 87417,c1(C(=O)NCCCCCNC(c2cc(O)cs2)=O)ccc2n[nH]cc2c1F 87418,C1(NC(C2(C)CCSCC2)=O)CC2CCC1N(C(c1ccc(F)cc1N)=O)C2 87419,C(CCCCCO)NC(CC(C)N(C(CN1CCC(C)C1)=O)C)=O 87420,C(=O)(C(C)C(C)c1ccc(F)cc1)N(CCNC(=O)CCc1ccc(Cl)s1)CC 87421,CN1CCOC(C(=O)NC(CC(=O)N(CCCO)CCCO)C2CC2)C1 87422,Cc1cc(S(=O)(=O)NC(=O)CC2CSC3CCCC23)c(Cl)cc1F 87423,N1(C(C#CC2(CC)CC2)=O)CCCN(C(c2cccc(C3CCC3)c2)=O)C(C)C1 87424,C12(C(=O)NC(C#C)CC(C)C)CCC(NC(C3CC34CCCCC4)=O)(CC1)C2 87425,Cc1cc(Cl)cc(C(N2CCCC(NC(c3cncc(O)c3Cl)=O)C2)=O)c1C 87426,CN1CCOC(C(=O)NCC(O)CCNC(c2cnccn2)=O)C1=O 87427,c1(CC)ccsc1C(=O)NC(C1CC1C(=O)N(C(CO)C(C)C)C)C 87428,Cc1ncc(N)cc1C(N1CC(C(C)NC(c2nc(Cl)c(Cl)s2)=O)C1)=O 87429,c1(C(N(CCCCNC(C(CC)C(C)(F)F)=O)C)=O)noc2c1CC(C)CC2 87430,C=CCCC(F)(F)C(=O)N1CC2CCC(C1)C2NC(C1CCCN1C=O)=O 87431,c1(CCC(=O)NCC(C(C)C)NC(C2(C(N)=O)CC2)=O)cncc(F)c1 87432,c1(CC(N2CCC(C(C)NC(c3nc(C)sc3)=O)C2)=O)ccc2c(c1)ncn2C 87433,c1(OC)cc(NC(=O)COC(c2nc[nH]n2)=O)cc(OC)c1OCCN1CCCC1 87434,C(=O)(C(C)(C)C(N)=O)N1CC(NC(C2C(C)OCCC2)=O)C1 87435,CN1CCN(C(=O)C(O)CCN(C)C)CC1CNC(=O)C1=CCC1.N12CCC1C2=O 87436,c1(SCC(=O)NC2CCN(C(CC(CCC)C)=O)C23CC3)nnc2ccccn12 87437,c1(C(=O)NCCN(C(=O)C(C2CCC(=O)N2)C)C(C)C)ncc(F)cn1 87438,Cc1cc(=O)n(CC(=O)OCCCC2CCC(C)(C)CC2)cn1 87439,C1(NC(C=CCC)=O)CCC12CN(C(=O)C(CC)NC(=O)OC(C)(C)C)C2 87440,N1(C(c2c(COC)n(C)nc2)=O)CCCN(C)C(=O)C1 87441,Cc1cccc(C(F)C(=O)N(CCCCNC(c2nn(C)cc2Cl)=O)C)c1 87442,N1(C(C(C)(C)OC)=O)Cc2occ(C(=O)NC3CN(C)CC3(C)C)c2C1 87443,C#CCCCC(C)C(=O)N(CCN(C)C(C1(C)COC(C)(C)CO1)=O)C(C)C 87444,C(CCCCCNC(C1CCC(C#N)C1)=O)NC(c1ccn(C)n1)=O 87445,n1(CC)ncnc1CN1CC(C(C)NC(C2CCCCS2)=O)C1 87446,CC1CN(C(=O)C=Cc2ccncc2)CC(C(=O)NCc2ccon2)O1 87447,c1(C(C(=O)NC2CC(CCNC(C(C)=CC)=O)C2)O)ccnn1C 87448,Cn1cc(C(=O)NC23CCCC(NC(=O)C(F)C(F)(F)F)(C2)C3)ccc1=O 87449,CN1CC=C(C(=O)NCC2(O)CC(C(=O)NC(Cc3cnc[nH]3)CO)C2)C1 87450,C(=O)(CCCCNC(=O)OC(C)(C)C)N(C(C(C)CC1CCCO1)=O)C1CCC1 87451,c1(C(N2CCC(O)(CN(C(C3C(CC)N(C)CC3)=O)C)C2)=O)cc(O)ccc1C 87452,N1(C(c2cccc(C#C)c2)=O)CCCC2(NC(C3CCCCC(=O)N3)=O)CC2C1 87453,Cc1cc(C)n(C(C)CC(=O)N(C)CC2CCN(C(c3ccc(F)o3)=O)C2)n1 87454,C1(NC(C(C)CO)=O)C2CC3C1C3C2C(=O)Nc1cc(O)cc(F)c1 87455,Nc1c(C(N2CC(NC(=O)Cn3ncnn3)CC(F)(F)C2)=O)ccc(Cl)c1Cl 87456,S(=O)(=O)(c1c[nH]ccc1=NCc1ccc2occc2c1)NC(c1cc(C)on1)C 87457,C1(C(N(CCCCCC)CC(N)=O)=O)CCC(CC2CCCN2C(C)=O)CC1 87458,C(=O)(C(C)(C)C(C)(F)F)N1CC2C(CC(=O)N(C3CCC3(C)C)C)C2C1 87459,N1(C(C2(SC)CC2)=O)CCC(C)C(NC(=O)C(C)(c2ccccc2)OC)C1 87460,C(=O)(C(CC)C(C)(C)CC)N1CCCC(N(C(CCCC(=C)C)=O)CCO)C1 87461,C(CC(C)C)(C(C(=O)Nc1ccc2c(c1)OCO2)N1CCC(C(N)=O)C1)OC 87462,c1(OC)cc(C)c(CN(c2cc(NCC(C)CC3CC3)nc(C)n2)C)cc1C 87463,S(=O)(=O)(c1ccc(Br)s1)N1C(C(=O)Nc2cc(C(C)(C)C)no2)CCCC1 87464,C(=O)(C(CC(C)C)NC(N)=O)NCC(=O)NCC1(CC)CC1 87465,CCCCCC(O)C(=O)NC1(CCC(=O)N(C(CO)C2CC2)C)CCC1 87466,CN1CC2C(CCCN2C(=O)NC2CCCN(c3ncccn3)C2)C1=O 87467,CC1(C)CCC(C(=O)NC(CCO)C2CCCC2)CN1C(C1(O)CCCC1)=O 87468,CCC(C)(COC)C(=O)NC1CC1CNC(=O)Cc1nn(C(C)C)cc1Br 87469,C(=O)(C=C1SCC(=O)N1C)N(CCC(C)NC(=O)CC1CC(=O)NC(=O)C1)C 87470,C1(CNC(C(C)C)=O)CN(C(C2CCCN(S(C)(=O)=O)C2)=O)CCCO1 87471,N1(C(C(C)C)=O)CCCCC1C(C)(C)CNC(c1ccc(N(C)C)cn1)=O 87472,C1(F)(CNC(C(C)OC)=O)CN(C(=O)CCNC(c2ccsc2)=O)C1 87473,N1(C(=O)Cn2cc(SCC#N)nn2)CCN(Cc2cc(C)on2)CC1.C1(=O)CN1 87474,c1(OC)cc(CNC2CCN(c3ccc(Cl)c(F)c3)C2=O)c(Br)c(C)c1 87475,C1(NC(C(CCC)C)=O)CN(C(C2CC(c3ccc(O)cc3)C2)=O)CCC1(C)C 87476,c1(C(=O)NC(CC)(C)CNC(C2CCC(C(N)=O)O2)=O)ccc(C2CC2)cc1 87477,C1(C(N(C(C#C)(C)C)C2CC2)=O)CN(C(=O)CC=Cc2ccccc2)CC1(C)C 87478,c1(C(=O)NC2(CC=C)CCN(C(=O)C=CCN(C)C)CC2)nc2ccc(Cl)nn2n1 87479,C=C=CC(C)C(=O)NCC1CCCN(C(C2(C)COC(=O)N2)=O)C1 87480,c1(C(N2CC(COC)(NC(=O)CSC(F)F)C2)=O)noc2c1CN(C(C)=O)CC2 87481,O=C(C1=CCCCCC1)NC(c1nnnn1CCCNSC1OC(=O)CC1O)C1CC1 87482,CC(C)S(=O)(=O)CC(=O)NC1CCN(C(C2CCCCCS2(=O)=O)=O)CC1O 87483,c1(C(N2CCC(C(=O)Nc3ccc(C4CC4)cc3)(CF)C2)=O)cccc(Cl)c1 87484,Cc1cc(CC(=O)N(C2CCCN(C(c3cnc(C)n3C)=O)CC2)C)ccc1Cl 87485,c1(C2(CNC(CCc3cccc(C)n3)=O)CCC2)c(F)cccc1F 87486,CC(C)CCCC(=O)N1CCC(NC(=O)C=CC2CCCCC2)C(O)C1 87487,CC(C)C(C)(CNC(C1CCC(=O)C1)=O)NC(c1ccc(C2CC2)nn1)=O 87488,C1(C)(C(=O)NCCC2(C(N(CC(C)OC)C)=O)CCC2)CCCOC1 87489,c1(C2N(C(c3ncccc3Br)C(=O)NC3COC3)CCC2)ccc2nonc2c1 87490,Cc1nnc2c(C(N3CCCN(C(=O)C(F)n4ccnc4)CC3C)=O)nccn12 87491,O=C(CC1NC(=O)c2ccccc21)NCCC1CCN(C(C2SCCS2)=O)C1 87492,C(CCC(C)CC(=O)N(C)CC1(NC(=O)COCCCF)CC1)=C(C)C 87493,c1(COC(C(COC)C)=O)cc(Br)ccc1C(=O)OC 87494,N1(C(CNC(CC(c2c(C)n[nH]c2C)C)=O)=O)CCOC(C)(C(F)F)C1 87495,N1(C(C(CC#C)O)=O)CC(NC(c2ccn(C)c(=O)c2)=O)CCC1C 87496,CC(CN=c1[nH]cnc2c(C(F)(F)F)cccc12)N(C)C(c1ccc(C2CC2)o1)=O 87497,N1(C(C(C2CCOC2)NC(Cn2ncc(C)c2)=O)=O)CCCC2(CC1)CC2 87498,C(=O)C1=CC2C=CC(C1)C2.N1(N2CCC(CC)C2COC)CCCC(C)(C=O)C1 87499,C(C)(CCS(C)(=O)=O)NC(NCCS(=O)(=O)NCC)=NCC1CCCCC1 87500,c1(C(C)(C)C)cccc(NC(=O)CC2CCC(C(=O)NC3CC(O)C3)CC2)n1 87501,C(=O)(C1Cc2ccc(F)cc21)NC1(C)CC(NC(CC(C)c2cccnc2)=O)C1 87502,Cc1cccc2nc(NC(=O)CC3CCCN3C)[nH]c12 87503,N1(C(C2N(C)CCOC2)=O)C2CCC1CN(C(c1ccc(C(F)F)c(F)c1)=O)C2 87504,N1(C(C)=O)CCC(CC(=O)NCCCN(C(c2cncn2C)=O)C(C)C)C1 87505,C=CCCC(=O)N(CC(C)NC(c1cscc1Cl)=O)CC 87506,C1(NC(C(C)OCC(C)C)=O)COCC1NC(c1nscc1Br)=O 87507,N1(C(C(C(C)O)C)=O)CCCCC(NC(=O)CCc2ccsc2)C1 87508,C(CC(CC)C(=O)NCC(C)(C)CNC(c1scnc1COC)=O)=CC 87509,C#CCCC(=O)NCCCN(C(=O)CC12CC(C(=O)OC)(C1)C2)C 87510,c1(OCC(=O)N(CCNC(C2(CC(C)C)CCCC2)=O)C2CC2)cccc(O)c1 87511,Cc1nc2ncnn2c(NC2CC3CC(C2)N(C(=O)CC2CSCCS2)C3)c1C 87512,c1(NCC2(CNC(=O)CCc3cc(Cl)cs3)CC2)ncnc2cc(C3CC3)nn12 87513,C12(C(N(C(C)CCNC(C3CC4(CCO3)CC4)=O)C)=O)CC3CC1C2C3(F)F 87514,c1(CC)nc(C(N2CCCC2CNC(=O)C=CCOC)=O)c2ccccn12 87515,CCC(F)(F)C(C)(C)C(=O)NC1CN(C(=O)C=C(Cl)Cl)CCC12CCC2 87516,C(CN=C(NCC(c1cccc(Br)c1)C)N1CCC2(CCOC2)C1)OC 87517,C1(COC)CC(CNC(=O)C=C2CCSCC2)N(C(=O)CSCCC(F)(F)F)C1 87518,c1(NC(C2CC(=C)C2)=O)cccc(C(N2CCOC(C(=O)N(C)C)C2)=O)c1 87519,C1(C(F)(F)F)(C(=O)NCCC(C)NC(C2OCCC2C(F)(F)F)=O)CC(F)(F)C1 87520,c1(C(C)C)nc(NCCC(C)OC(F)F)cc(=NCC=O)[nH]1.C(C)(C)(C)O 87521,C(=O)(C1=C(SC)CCCC1)NCC1CCN(C(c2c(CC)csc2)=O)CC1C 87522,C1(OC)(OC)CCN(Cc2ccc(Cc3ccccc3)cc2)CC1O 87523,c1(C(N2CC(C(=O)NCC3C(C)C3C)C(F)C2)=O)cccc(C#N)c1 87524,c1(SC)ncc(C(=O)NC2CN(C(C3CCC(C)(C)CO3)=O)CCC2C)c(O)n1 87525,C1(OC)CCCCN(CC(=O)NCC(C)N(C)C(C2C(C)(C)OC2(C)C)=O)C1=O 87526,N1(C(CCCC#CC)=O)CCC2(CC1)CC(NC(=O)CSC)CCO2 87527,Cc1cc(=NCC(=O)Nc2nccs2)[nH]c(=NCC2CN3CCCCC3CO2)[nH]1 87528,C1(CNC(C2(C)CCC2)=O)C2CN(C(=O)CCc3cccs3)CC12 87529,C1(C(=O)NCC(CN(C)C)(C)O)CC(=O)N(c2cccc(Br)c2)C1 87530,N1(C(CN2CCC(N(C(C(C)C)CO)C)C2)=O)CCCN(C(=O)CO)CC1 87531,CC1=C(C(=O)N2CC(NC(c3ccc(C(N)=O)c(Cl)c3)=O)C(F)C2)CCO1 87532,C(c1cc(Cl)c2c(c1)OCO2)=CC(N1CCC(C)C(NC(=O)C(C)N(C)C)C1)=O 87533,C(c1ccc(C#N)cc1)=CC(=O)NC1(CNC(C2CC(C)OCC2)=O)CC1 87534,Cc1cc(O)cc(C)c1C(N1CC(F)(CNC(C2(C)CC3CC3C2)=O)C1)=O 87535,C(=O)(C(C)(C)CC(C)C)N1CC(C(N2CCC(C=C)(O)C2)=O)OC(C)C1 87536,C1(NC(CC2ON=C(C)C2)=O)CCCCN(C(C2CC(N(C)C)C2)=O)C1 87537,C(N=c1cccc(S(=O)(=O)NC2CC(F)(F)C2)[nH]1)c1ccc(C(C)OC)o1 87538,N1(C(=O)NC(C2CCC2)C2CC2)CCC2(CC1)CC2(C)Cn1c(C)ncc1 87539,Cc1cc(Cl)c(C(N2CCC(O)(C(C)NC(c3cccc(F)n3)=O)C2)=O)cc1C 87540,c1(OC)cc(C(N2CCOCC2CC(=O)Nc2cc(C)cc(O)c2)=O)ccc1O 87541,c1(CC(N2CCC(CNC(c3ccco3)=O)CC2)C)ccc(Br)cc1 87542,C1(c2nc(C3C(F)(F)C3C(F)(F)F)on2)CC2(C1)CC21CCC1 87543,CC1(C)CC(CO)CN(C(CCc2ccccn2)C(=O)NCCC2(C)CC2)C1 87544,N1(CC#C)CCN(C(C2CSCN2C(=O)CCc2cnoc2)=O)CC1=O 87545,c1(C(N(CCCOCCN(C(CN2CC(C)(OC)C2)=O)C)C)=O)cc(Cl)ccn1 87546,C(=O)(C#CC(C)(C)CNC(=O)C(F)C1CCC1)NC(c1ccc(C)cc1)C 87547,N1(C(C(C)OCC#C)=O)CCN(C(c2cnn(CC)c2C)=O)C2CS(=O)(=O)CC12 87548,C1(NC(c2cc(OC)c(O)c(Cl)c2)=O)CN(C(C2CCC2)=O)C2(CCCOC2)C1 87549,C(=O)(CCCCC(N)=O)NC1(C)CCN(C(=O)C=Cc2ccccc2)C1 87550,C1(NC(C2C(=C)CC2)=O)CCC2(CC1)CN(C(=O)CCC(=O)OC(C)(C)C)C2 87551,N(C)(C1CCc2cc(F)ccc21)C(COc1cccc(C(=O)OCC)c1)C 87552,C(COC)(CC(=O)NCC1(CC)CC1)NC(C(C)=CC=C)=O 87553,c1(C(N2CCCC(C)(NC(C(C)=C3CCCC3)=O)C2)=O)ccn2cc(C)nc2c1 87554,C1(F)(C(N2CC(NC(C(CC)C(C)C)=O)C3(C2)CC3)=O)CCC(F)(F)CC1 87555,c1(N2CCCN(CCC)CC2)nc(=NCc2cnn[nH]2)[nH]c2cc(C)ccc12 87556,CCCCC(O)CC(=O)NCC(C1CCCC1)NC(c1ncccc1Cl)=O 87557,C1(n2cc(CN(CC(C)(C)OC)C)nn2)CCCCCC1O 87558,N1(C(CCC(C)OC)=O)CC2CC1CCC2NC(=O)CC1CCCCC1O 87559,C(=O)(CC(C)(C)C(F)F)NC(CCCC)CNC(c1cc(C2(O)COC2)on1)=O 87560,C(c1cn(C)cn1)=CC(=O)NC1(CC)CN(C(C2C(OCC)CCC2)=O)C1 87561,Cc1nc[nH]c1CC(=O)NCC1(CCNC(c2cc(C(F)F)cs2)=O)CC1 87562,c1(C(N2CC(C)C(n3cc(CCC4CC4)nn3)C2)=O)cccc2ncsc12 87563,Cn1c(O)ncc(C(=O)NC(c2ncon2)Cc2ccccc2)c1=O 87564,c12ncc(F)c(n1)N2C(=O)COCC.C1(SC)CCCNC1 87565,C#Cc1ccc(CC(N2CCC(NC(c3c(C)csc3Cl)=O)C(CO)C2)=O)cc1 87566,c1(OC)ccnc(C(N2CC(O)(CCNC(=O)C(C3CCOCC3)C)C2)=O)c1F 87567,C1(C(=O)NC2C(NC(c3cc(C(C)C)[nH]n3)=O)C2)CCC(C(F)(F)F)CC1 87568,N1(C(c2cc(C)ncn2)=O)CCN(C)CC1CNC(c1ccoc1CC(N)=O)=O 87569,c1(C(N2C(CN(C(C3CN(C)C3)=O)CC)CCC2)=O)cccc(O)n1 87570,Cc1cnc(NC2(C)CC2)c(S(=O)(=O)NCCC(C)c2cn[nH]c2)c1 87571,c1(OC)cc(C(=O)Nc2cccc(N(C)C)c2)c2ccccc2c1 87572,C1(CNC(N(CCCN(C)C)C)=O)CCN(C(=O)C(C)(C)C)CC1.C1CO1 87573,c1(CCC)cc(=NC(CNC(c2coc(CCOCC)n2)=O)C2CC2)[nH]c(Cl)n1 87574,c1(CNC(=O)CCC2CC2)ccc2c(c1)CCC2NC(c1cccc(O)n1)=O 87575,C=Cc1cncc(C(N2CC(O)(C(F)C(=O)NCC(c3ccncc3)O)C2)=O)c1 87576,N1(C(CC(CC)SC)=O)CCC(O)C(NC(=O)CCC(C)C)C1 87577,C(=O)(CC(C)(C)N(C)C(C1(CO)CCCCO1)=O)NC(C#C)C1CC1 87578,CC(CN1CCCC1=O)N=c1cccc(S(=O)(=O)NCc2c[nH]nc2C(F)F)[nH]1 87579,C(=O)(CC1=CCN(CC2(C)CCCN2C(C)=O)CC1)OC 87580,c1(OC)cc(C(=O)NC2CCC(NC(C3CC(CF)C3)=O)C2)ccc1C 87581,Cc1sc(C(=O)NCCC2CCN(C(=O)C(=O)CC(C)C)C2)cc1[N+](=O)[O-] 87582,N1(C(C2(CC)CCCCC2)=O)CCC(C)N(c2nccc(CC(C)C)n2)CC1 87583,c1(OC)ccc2nc(S(C)=O)[nH]c(=NCc3cnn[nH]3)c2c1 87584,c1(CCN(CCN2CCN(C(=O)OC)CC2)CC)ccc(Cl)cc1Cl 87585,C(=O)(C(C)(C)CS(N)(=O)=O)N1CC(NC(C(C2CC2)OC)=O)C(C(F)F)C1 87586,Cn1cncc1C=CC(=O)NCC(C1(O)CN(C(C2C3CNC(=O)C23)=O)C1)(C)C 87587,Cc1ccc(NC(C2CC(C)N(C(c3cnn4c3CCC4)=O)C2)=O)cc1C 87588,C#Cc1cnn(C)c1C(=O)NCC1COCCN1C(C1C2CCC1CC2)=O 87589,C1(NC(c2cc(Cl)ccc2F)=O)CN(C(=O)CCCC(F)F)CC1C1CC1 87590,c1(C(N(C2CC(NC(C(C(CC)CC)C)=O)C2)C)=O)cnn2cccc(OC)c12 87591,CN1CCc2ccc(C(=O)NCC(CO)NC(=O)C3=NNC(=O)CC3)cc21 87592,CCC(C)C(C(=O)NCC1CN(C(C23CC(C)(C2)C3)=O)CC1C)OC 87593,C(=O)(C(C)CC(F)(F)F)NCC1CN(c2cc(C)nc(C(C)(C)C)n2)CC1(C)C 87594,C(=O)(CCS(C)(=O)=O)NC1(C(=O)NC(CC)CN2CCCC2)CCSC1 87595,c1(C(=O)NC2CC(NC(=O)C=Cc3cc[nH]n3)C2)ccc(C2CC2)nc1 87596,N1(C(c2c(C)n(C)cc2)=O)CCC(NC(=O)C(O)C(F)F)C2(CCC2)C1 87597,c1(OC)ccc2nc(OC)[nH]c(=NCC3OCCc4sccc43)c2c1 87598,N1(C(c2c(C)n(C3CCOC3)nn2)=O)CCC(CNC(C2CC2(Cl)Cl)=O)C12CC2 87599,c1(CC(=O)NC2CC2NC(c2csc(-c3ccccn3)n2)=O)ccc(O)cn1 87600,c1(C(=O)OCC)ccn(CC(=O)NCCC2CC(NC(=O)CC3CCOC3)C2)n1 87601,O=C(C1=CS(=O)CCC1)NCCN(CCOCCO)C(C1(OC)CCC1)=O 87602,O=[N+]([O-])c1ccc(Br)c(Cl)c1NCc1nccs1 87603,c1(CC=CC)ccccc1C(=O)NCC(C)CNC(c1snnc1C1CCC1)=O 87604,Cc1cc(N(CCC(N)=O)C)nc(N2CC=CCC2)n1 87605,N1(CCC(=O)NCC2CC(O)CN2C(=O)COC2CCCCC2)CCOCC1=O 87606,C(N=c1ccnc(C)[nH]1)C1CCCC(NC(C(c2cc(C)c(F)cc2)(C)C)=O)C1 87607,c1(C(=O)NC2C3(CN(C(C4(CC)COC4)=O)C3)CC2)coc(S(=O)(=O)NC)c1 87608,N1(C(C(c2ccc(OC)nc2)(F)F)=O)CCC2(NC(=O)CC(C)(C)O)CCCC12 87609,N1(C(c2cc(C)c(C)s2)=O)CC2(CC(NC(=O)CS(=O)(=O)N(C)C)C2)C1 87610,N1(C(=O)C=Cc2ncc[nH]2)CC(CO)C2(C1)CN(C(c1cc(Cl)cnn1)=O)C2 87611,C1(NC(CCCNC(=O)NCC#C)=O)CN(C(=O)CS(=O)(=O)N(C)C)CCC1C 87612,c1(OC)ccc(OCC(CP(C)(C)=O)OC(CCNc2ccc(F)cc2)=O)cc1 87613,O([Si](C)(C)C(C)(C)C)CCCOC(C1(CC(C)C)CC(=O)C1)=O 87614,CCC(CNC(=O)C(C(=O)OC)OC)(CC)C(=O)Nc1ccc(O)cc1Cl 87615,C(=O)(C#CC1(C(F)(F)F)CC1)NC1C(CNC(CCCN(C)C)=O)CCC1 87616,N1(C(c2c(CC)ncs2)=O)CCCC2(C1)CN(C(c1cccc(C)c1Cl)=O)C2 87617,CC1CN(C(=O)CS(=O)(=O)NC(C)(C)C)C(C)CN1C(c1cnn(C(F)F)c1)=O 87618,CN1CCN(C(C2CC(C3CC3)=NO2)=O)C(C(=O)NC2(CCF)CCC2)C1 87619,CCCCN=C(NCCc1ccc(Cl)c(Br)c1)NCCc1cccs1 87620,C1(C)(C(N(C2CCN(C(=O)CCCCNC(N)=O)CC2)CC#C)=O)CCCCC1 87621,c1(C(N(C2CCCCN(C(C3(C)CC=CC3)=O)C2)C)=O)cc(Br)cnc1O 87622,N1(C(COCCCC#C)=O)CCCCC1C(=O)NCc1cnc(OCC)cn1 87623,c1(OC(CS(N2C3CN(C(C)=O)C(C3)C2)(=O)=O)=O)cc(CO)c2ccccc2c1 87624,C1(C)(CNC(CN(C)C(=O)C2CC2)=O)CCN(C(C2C3CNC(=O)C23)=O)CC1 87625,N1(C(c2c(CNC(c3c(C)nccn3)=O)c[nH]n2)=O)CC2NC(=O)OC2C1 87626,C1(NC(C(CN(C)C)(F)F)=O)CC2(C1)CC(CNC(c1ccc(Cl)c(F)c1)=O)C2 87627,c1(C(C(=O)N(C2CCC2)C(C)=O)N(CC(F)F)CCC)sc(Br)c(C)c1C 87628,c1(C(=O)NC2C(NC(C(C)(C)C3CCCO3)=O)COC2)cc[nH]c2nccc1-2 87629,C(=O)(C#CC1CCCOC1)NCC1(C)CCN(C(c2c(N)ccc(CC)c2)=O)C1 87630,C12(C(N3CCC(NC(C=C(C)Cl)=O)C3)=O)CCOCC1C2 87631,C(C1CN(C(=O)C(O)CC2CCCC2)CC1C(=O)NCC(C)C(C)C)=CC 87632,Cc1cccc2[nH]cc(CN3CC(F)CC3C(=O)NC3CCCCC3O)c12 87633,c1(CC)c(C(N2CCCC2C(C)(C)C(=O)NCCn2cccn2)=O)ccn1C 87634,N1(C(C=CCCC)=O)CC(NC(c2ccc(OC)s2)=O)CCC1C 87635,C1(CC(=O)NC2CCN(C(C)C)C2)(OC)CN(C(=O)CC2CC(F)(F)C2)C1 87636,N1(C(CCC2(C)CC2)=O)CC2CC1C2C(=O)NCC1CC(F)C1 87637,C1(C(N2CCC(C(=O)N(C)CC3CC3)(OC)C2)=O)Cc2nccn2C1 87638,c1(CC=CCNC(c2[nH]cc(CC(C)C)c2)=O)nc2c(cc1C#N)CCC2 87639,C1(C(=O)NC(CCCCNC(CNC(=O)OC)=O)(C)C)COc2ccccc2C1 87640,c1(C(=O)NC2CN(C(CSCC)=O)CC2(C)C)sc2ncccc2c1Cl 87641,N#Cc1cccc(OCC(=O)NCCCCNC(=O)CC2CCC(F)(F)C2)c1 87642,CC1(C)OC(=O)CC1C(=O)NC1(CCCNC(=O)CCN2CCC2)CC1 87643,C(=O)(C(F)(F)C(F)(F)F)N1CC(CN(C)C(c2cnn3cc[nH]c23)=O)C1 87644,c1(C(=O)NCCC(CNC(C(CCC)N(C)C)=O)O)c(C)nc(=N)[nH]c1C 87645,C1(CC(=O)NCCNC(c2nc(C)sc2)=O)CCCC(C)C1 87646,C(CC1=CCN(C(c2cccc3c2NCC3)=O)CC1)NC(CC1C(C)CCO1)=O 87647,c1(C(=O)NCc2ncc(C(C)C)cn2)cc(Cl)c(Cl)cc1Br 87648,N=S1(=O)CCCC2(CCCN2C(=O)CC(N)Cc2ccc3ccccc3c2)C1 87649,CCC(C)(O)C(=O)N1CCCC1c1nc(C(N2CC(C(=O)OC)C2)=O)cs1 87650,C1(OC)CCCN(C(C2(NC(=O)CC(C)F)CC(F)(F)C2)=O)CC1 87651,N1(C(c2c(C)noc2C)=O)CCC2(CC1)CC2C(=O)Nc1c(C)ncnc1C 87652,C1(COC)C=CCCN1C(c1occc1CNC(c1c[nH]cc1C)=O)=O 87653,C1(NC(c2cc(C(C)C)[nH]n2)=O)CCC2(CC1)CN(C(c1cncc(F)c1)=O)C2 87654,N1(C(c2c(CNC(C3(C(=O)OC)CC3)=O)cco2)=O)CC(C)CCCC1C 87655,N1(C(C)=O)CCCC1C(=O)NC(C)CCCNC(=O)C(O)CC1CCCCC1 87656,Cc1cc(C(=O)NCC2COC(CNC(c3cnn(C(C)C)c3)=O)C2)nn1C(F)F 87657,N1(C(c2cncc(N(C)C)c2)=O)CCOCC(NC(C2CC=CCC2)=O)C1 87658,N1(C(CC2(OC)CCCC2)=O)CCN(C(=O)CCN2CCC(O)CC2)C(CF)C1 87659,N1(C(C(C)=C2CCCC2)=O)CCN(C(c2cc(-c3ccccc3)no2)=O)C(C)C1 87660,Cc1nc(NCCCCC(N)=O)cc(=NCC2CCC(=O)NC2)[nH]1 87661,N1(C(c2oc(C)c(Br)c2)=O)CC(C)CN(C(=O)C(F)=C2CCC2)C(C)C1 87662,N1(C(C2(C#C)CCC2)=O)CC2COCC(C1)C2NC(C12CCCN(CC1)C2)=O 87663,C(CC(C(C)C)NC(=O)OC(C)(C)C)NC(C1CCCCC1)CC 87664,c1(C(=O)NCC(CCC)NC(c2ncccc2O)=O)cccc2nccn12 87665,C(C(C)(C)CC1CCC1)N(C(C)(C)C)C(c1nnnn1C1CCOCC1)C1CC1 87666,c1(C(=O)NC2C(NC(C3(CCOCC)CCC3)=O)C2)cnc2c(c1)NC(=O)CO2 87667,c1(C(=O)NCC2CCCCN2C(=O)CC2CCCCO2)cncc2nc[nH]c12 87668,CCCCCCOC(C)C(=O)NCCC1(CNC(c2cnc(N(C)C)s2)=O)CC1 87669,N1(C(c2cnc(OC)s2)=O)CC2CC1C2NC(=O)Cc1sc(C)nc1C 87670,Cc1cc(CO)ncc1-c1sccc1SC.C1N2CCCC2C1.c1ccnn1C(C)C 87671,N1(C(CCC=CCC=C)=O)CC=CC(C(=O)NCc2ccccc2C)C1 87672,c1(C(=O)NC2CN(C(C(c3ccncc3)C)=O)CC2(C)C)cc2c(o1)CCCC2 87673,c1(C(=O)NCC2(C)CCN(C(CCCCCSC)=O)C2)cc2nc[nH]c2cc1F 87674,CC(C(C)(C)C#N)NC(C1C2CC1N(C(C1C3CC(=O)CC13)=O)C2)=O 87675,CCCCC(C(=O)OC(C)(C)C)NC(=O)NCc1cc(CCCOC)cs1 87676,Cc1cc(C(=O)N(CC(O)CNC(c2ocnc2C(F)(F)F)=O)C)sc1Cl 87677,C1(OC)C2CC3CC1CC(C(=O)Oc1ccccc1)(C3)C2.N12CCN(CC1)CC2 87678,C(CCCCn1cc(Cn2ccnc2C)nn1)NC(C1(CCC)CC1)=O 87679,N1(C(CC2(CNC(=O)CC3CCCC34CC4)CC2)=O)CC2CCCC(O)C2C1 87680,CC1CC(NCc2nn(C)c3c2COCC3)c2ncnn21 87681,N1(C(C2CCN(CC)C2)=O)CCC2(C(=O)NC(CO)CC(C)C)CCCC12 87682,n1(CC(=O)NC2C3(CCN(C(C(C)C4CC4)=O)CC3)C2)[nH]cc2c(=O)ncnc1-2 87683,C1(O)(CNC(CCC(C)NC(c2ncnc(O)c2F)=O)=O)CC2C=CC1C2 87684,CC1(C)CC(CC(N2CCC(CF)(NC(c3cc([N+](=O)[O-])n[nH]3)=O)C2)=O)NC1=O 87685,c1(CN(C(C(CN(C(C)C)C)N)=O)C)ccccc1N 87686,N1(C(CCCOCC=C)=O)CCC2(CC1)CCN(C(c1ccc(Cl)c(O)c1)=O)C2 87687,N1(C(C(CC=C)CNC(=O)C(C)(O)C2CCC2)=O)CCOCC2(CCC2)C1 87688,C12(NC(C3C(COC)C3)=O)CCC1CN(C(c1ccc(Cl)cc1Cl)=O)C2 87689,C(CCC(C(=O)NCC1(F)CC1)NC(=O)Cc1cncnc1O)OC 87690,CC(CC(=O)N(C)Cc1cn(Cc2conc2C2CC2)nn1)c1cnn(C)c1 87691,CC(C)C(C)C(=O)NC1(CCNC(=O)Cc2coc(-c3ccccc3)n2)CC1 87692,CN1CCCC(O)(CC(=O)NCC2(F)CN(C(c3cccc4nonc34)=O)C2)C1 87693,C1(NC(=O)CC(F)(F)F)CC2CCC(C1F)N2C(C1(Br)CC1(F)F)=O 87694,C1(CNC(C)=O)CCC(F)(CNC(=O)C(C)CCN(C)C)CC1 87695,c1(C(N2C3(CNC(C(C)=CC)=O)CCC3CC2)=O)ccc2ccccc2n1 87696,C(=O)(CCCN(C)C)N(C1CCC(NC(C2(F)CCC2)=O)C1)C 87697,C1(F)(CNC(C(COC)OC)=O)CCC(CNC(=O)C(c2cnccn2)C)CC1 87698,C1(NC(c2ccc(OC)s2)=O)C(C)CN(C(c2cn(CCO)nn2)=O)CC1C 87699,C1(NC(c2ccnc(F)c2Cl)=O)CCN(c2ccnc(Br)n2)CC1F 87700,N1(C(C)=O)CCCC(CCNC(c2sc(F)cc2C)=O)CC1 87701,C(C(=O)N1OC2CCC1C2)C1(C)N(CC)CCC1.C1CCCC(=O)N1 87702,CC1=NS(=O)(=O)NC(C)=C1CCC(=O)NC(C1CCCCN1C(=O)C=C1CC1)C 87703,N1(C(C=C2CCC(C)C2)=O)CCCN(C(=O)Cc2cncc(Br)c2)CCC1 87704,N1(C(c2ncn(C(C)C)n2)=O)CCC2(CCC2NC(c2cnncc2O)=O)CC1 87705,c1(C(=O)NC(c2cnc[nH]2)C)coc(CNC(c2ccsc2Cl)=O)n1 87706,Cc1cc(C(=O)NCCN(C(=O)Cc2cncc(C#N)c2)C2CC2)ccc1Cl 87707,O=C1CC(C(=O)NC23CCN(C(c4cccc(Cl)c4F)=O)CC2C3)CC(=O)N1 87708,c1(C(=O)NCC(C)CNC(=O)C(c2ccccc2)O)cc(Cl)c(Cl)cc1N 87709,C1(C(=O)OC)(CC(c2ccccc2)C2CC2)CCNCC1.C1(=O)C(C)CN1 87710,Cc1cn2cc(C(=O)NC3CCC3CNC(c3cnc(C(C)(C)C)s3)=O)nc2s1 87711,N1(C(C(CCC)O)=O)C2CCCC1CN(C(=O)C(O)C1CCC1)C2 87712,c1(C(=O)NCC2CCC(NC(CC3(C(=C)F)CCC3)=O)C2)ccc(C#N)c(C)c1 87713,N1(C(C2N(C(CC)=O)CSC2)=O)CCCC(O)(CNC(C23CCC(C2)C3)=O)CC1 87714,CCCCCC(C)(C)C(=O)NC(CO)CCCCNC(c1c[nH]nc1[N+](=O)[O-])=O 87715,C=CCC(C(=O)N1CC(N(C)C(c2ccn(CCC)n2)=O)C1)c1ccccc1 87716,C=CCCCCC(=O)N1CCC(C2CCCCN2C(=O)C(O)C=CCCC)CC1 87717,c1(OCC)cccnc1C(=O)NC1CCCC1NC(C1(C)CCC(=O)N1)=O 87718,CC(C)CCC(O)C(=O)NCCCCC1CCN(NCCOCCO)CC1 87719,c1(CCC)n[nH]c(=NC(=O)N2CC(C(N)=O)C(c3ccccc3)C2)s1 87720,N1(C(C(CC)Cc2ccccc2)=O)CCCC(C)(CNC(C2CC(Cl)(Cl)C2)=O)C1 87721,c1(CC(=O)NC(C)CNC(c2cncc(N(C)C)c2)=O)ccccc1S(C)=O 87722,C1(C(=O)NCCN(C(=O)CC(C)(F)F)CCOC)CCc2cncn2C1 87723,C1(NC(c2occ(C)c2)=O)COC2C(NC(=O)C(F)F)COC12 87724,C1(NC(=O)CCCc2cccs2)COC2C(NC(c3cn(CF)nn3)=O)COC12 87725,c1(CC)nc(C(=O)NCC2CN(C(=O)C(c3ccccc3)C)CC2O)c(C)o1 87726,c1(C(=O)NC2(CNC(c3n[nH]cc3F)=O)CCOC2)cnn2c1OCCC2 87727,c1(SCC)cc(C(=O)NCCC2(NC(=O)CC(CC)SC)CCCC2)ccc1F 87728,N1(C(C(C)O)=O)CC2CC1(CNC(=O)CC1CCCCC1F)C2 87729,C1(C(=O)NC2(CNC(c3occ(C)c3)=O)CCOC2)COC(C)(C)CO1 87730,C1(CCNC(C(C)(C)Br)=O)CCN(S(=O)(=O)Cc2cccc(Br)c2)CC1 87731,c1(CC)ccc(C(N2CC(CNC(=O)CCc3n[nH]c(=N)s3)C(C)C2)=O)c(F)c1 87732,C1(C(N(CCO)CC)=O)CC2CN(C(C3CCCCC3)=O)CC2C1 87733,CC1CN(C(c2ccc(C3CC3)nn2)=O)CCN(C(c2cnnn2C)=O)C1 87734,n1(CCC(=O)NC(C2CCOC2)CNC(C23CCC2CC3)=O)ccc(O)nc1=O 87735,N1(C(c2c(OCCC)cccc2)=O)CC(NC(=O)C(C)n2cccc2)CC(C)C1 87736,C=CCC(CC(C)C)C(=O)N1CCOC(CN(C(=O)CCc2cnn[nH]2)C)C1 87737,C1(NC(C2C(OC)CCC2)=O)CN(C(=O)C(Br)=C(C)C)CC(C)(C)C1 87738,c1(CC(=O)NCC(C)N(C(Cc2ccc(C)cc2)=O)C)nn(C)cc1[N+](=O)[O-] 87739,Cc1nn(C)c(=O)c(C(=O)NCCC2CCN(C(C3CCC(=O)N3C)=O)C2)c1C 87740,C1(NC(CCCCOCC)=O)CCN(C(=O)C(C)(C)C2CC2)CC1C 87741,N1(C(C2(C#N)C(C)(C)C2)=O)CCC(C=CC(=O)NC2CC(N3CCCC3)C2)CC1 87742,C1(C)(C(N(C)CC2CCCN(C(CC(=O)OC)=O)C2)=O)CCS(=O)(=O)CC1 87743,C1(O)(C(=O)NC2CCN(C(c3nc(COC)oc3)=O)CC2C)CN2CCC1CC2 87744,C(CN=c1[nH]c2c(c(=NCc3nc(C4CC4)cs3)[nH]1)CSC2)C1(CO)CC1 87745,C1(C(=O)NCCNC(C)=O)CN(C(=O)C(C)(C)COC(C)(C)C)CCCO1 87746,N1(C(C2C(CC)CCC2)=O)CC(NC(=O)CC(=O)NC2CC2)CC2(CCC2)C1 87747,c1(OC)ccccc1C=CC(=O)NCC(C)(CO)NC(c1cc(F)ccc1C)=O 87748,C1(C(=O)NCC(C(C)C)NC(c2cc(CO)on2)=O)CCC(C)CC1 87749,c1(C(N(CCNC(CSCCC#N)=O)CC2CC2)=O)ccc2ccoc2c1 87750,c1(OC)nc(NC(C2CC2NC(c2scc(C)c2Cl)=O)=O)cnc1C#N 87751,c1(CCNC(NC(C)Cc2ccccc2C(F)(F)F)=S)ccc2c(c1)OCCO2 87752,N1(C(C2(C)CCCCO2)=O)CC2CC(NC(=O)C(O)C3CC3)CC2C1 87753,C1(C(=O)OCC)CCN(C(=O)CCN(C(C2CC2N(C)C)=O)C2CC2)C1 87754,N1(C(CCC(C)(C)OC)=O)CC2(CCCN(C(c3cccc(C)c3C)=O)C2)C1 87755,C1(C(N2CCC(C)(CNC(c3nc(OC)c(C)s3)=O)C2)=O)CC(C)(C)C(C)(C)C1 87756,c1(N2CCC(OC)(CO)CC2)nc(NCC2(CF)CCC2)c2cnn(C)c2n1 87757,C1(N(C(CC(C=C)c2ccccc2)=O)C)CCCN(C(=O)C=CCN(C)C)CC1 87758,c1(C(c2nnnn2C2CC2)NC(CCC)CC)ccc(OC)c(F)c1F 87759,CC1CC(C(=O)NCc2nocc2C(=O)N(C)CC2CC(F)(F)C2)CCO1 87760,N1(c2nccc(C(=O)OC)n2)CC2(CCCC2NC(=O)CCC(C)C)C1 87761,Cc1cc2ccc(C(=O)NC3CCCCC3NC(C3CC3Br)=O)cn2c1 87762,Cc1cnc(NC2CC(NC(=O)Cn3nc(O)ccc3=O)C2(C)C)nc1O 87763,c1(C(N(CCNC(c2cccc(C)c2F)=O)CC2CC2)=O)ccc2nn[nH]c2n1 87764,C1(C(=O)Nc2n(CC(=O)OCC)ncc2)CN(C(C2(C)CCCCC2)=O)CCN1 87765,C1(C(=O)OC)CC(O)(CC(=O)NC2(CNC(C3(O)CC3)=O)CC2)C1 87766,N1(C(C(=O)NCc2nnn(C)n2)CCC2CCCO2)CCC(S(=O)(=O)C(F)F)C1 87767,c1(C(N2CC(C(N(C)CC3CCCC4CC34)=O)OCC2)=O)c(F)cccc1F 87768,c1(OC)cc(CN2CC(NC(c3ccoc3)=O)CC(F)(F)C2)cc(I)c1O 87769,C12(C(C)NC(c3coc(CNC(=O)Cc4cn(C)cn4)c3)=O)CCC(CC1)C2 87770,Cc1cccc(CCCNC(c2ccnn2C2CC2(F)F)c2nnnn2C)c1 87771,CCC(CC(=O)N1CCN(C(=O)CCc2ccc(C)s2)CC1COC)C(F)F 87772,c1(OC)cccc2c(CC(=O)NCCCN3CC(C)CC(C)C3)c[nH]c12 87773,Cc1cccc(N)c1C(=O)NCC1C(C)CCCN1C(=O)Cc1cccc(F)c1 87774,c1(CCC)onc(C)c1C(N1CC2CC2(C(=O)NCc2cccc(Br)n2)C1)=O 87775,c1(C(N2CCCC(OC(C)(C)C)C2)C(=O)NC(CC)(C)C)ccc2c[nH]nc2c1 87776,c1(C(N(CC(C)NC(c2cnc(C(C)O)s2)=O)C)=O)cnn(C)c1C1CC1 87777,C1(C(N(C2CCC2O)C)=O)CC(O)C(O)CC1CNC(=O)CC1(N(C)C)CC1 87778,C1(NC(C2CCn3ccnc3C2)=O)CCCC12CCN(c1nncs1)CC2 87779,Cc1cc(N)c(C(=O)NC(C2CN(C(c3cccc(F)n3)=O)CCO2)C)cc1F 87780,c1(C(=O)NC2CCCC(NC(=O)C3=CCC3)C2)ccc2c(c1O)CCCC2 87781,C1(CNC(C(CC#C)C)=O)CC2(C1)CN(C(=O)Cc1ccnc(C(F)(F)F)c1)C2 87782,c1(C(=O)NCC(C(C)C(C)C)NC(Cc2cnc(C)[nH]2)=O)cc2ccccc2o1 87783,c1(NCC(N2C(CN(C(C(CC)OC)=O)CC)CCC2)=O)ccc(C)cc1 87784,c1(OC)cc(OC)cc(C(=O)NCC(C)(C(C)C)NC(c2ccc(Cl)cc2)=O)c1 87785,C1(NC(CC(c2ccc(NC)cc2)C)=O)CCNCC12CC2 87786,CC(C(=O)NCc1cncs1)N(C(C1CCC1)=O)C1CC1 87787,C(C1=CCCN(C(C2C3CCCOC23)=O)C1)NC(=O)Cc1cnc(C2CC2)[nH]1 87788,c1(C(N2C(C)CN(C(C3CCC(=O)N3)=O)CC2)=O)ccnc(P(C)(C)=O)c1 87789,C1(CC(=O)NCCC(=O)N(CCn2c(C)ncc2)C)CCCCN1C 87790,c1(C(=O)NCC2C(C(=O)NCC(=O)N(C)CC)CCC2)ccccc1C1CC1 87791,C1(C(N2CCCC(NC(c3c(COC)cco3)=O)C2C)=O)CC2CCCCCCC12 87792,c1(C(=O)NC2(C(N)=O)CCOC2)ccc(CC#N)cc1.C1(=O)CCN1C 87793,c1(CCC(=O)NCC(O)COc2ccc3n[nH]cc3c2)cccc2c1OCCO2 87794,C1(C(=O)NCC2CC2C(=O)NOCC2CCC2)C=CCOC1 87795,N1(C(C2CCC(=O)N2)=O)CC2(CCCC2NC(c2ccc3ncsc3c2)=O)C1 87796,c1(CNC(C(C)(C)NC=O)=O)cccc(CNC(=O)C(F)(F)CN2CCCC2)c1 87797,C1(C(=O)NC2CCN(C(CC3C(C)(C)C(O)C3)=O)CC2F)CC2C=CCC(C1)C2 87798,N1(C(CNC(CC)=O)=O)CCC(C(C)NC(c2sc(C)nc2CC(C)C)=O)CC1 87799,C(=O)(C1=NOC2COCC12)N(CCNC(C(C)SC)=O)CC1CC1 87800,C=CCCCCC(=O)NC1COCC1CNC(c1c[nH]c(Br)c1)=O 87801,N1(C(c2occ(C)c2)=O)CC2OCCN(C(=O)CC3C=CCCC3)C2C1 87802,C(C1=CCN(C(=O)CC(C2CCC2)C2CCC2)CC1)NC(=O)CC(F)(F)F 87803,Cc1cc(C(=O)NCc2cc[nH]c2C(=O)NCC(c2cnc[nH]2)C)[nH]c1C 87804,c1(NC(C(=O)N(C2CC3CCC2C3)C)=O)cncc(SC(C)(C)C)c1 87805,N1(C(C(C(C)C)O)=O)CC2CN(C(=O)COCC3CCCCC3)CC2C1 87806,c1(OCCOCCOC)cccc(C)c1C.c12ocnc1CNC(=O)N1CC2C1 87807,C1(NC(CC(C)(C)C)=O)CC2(C1)CN(C(c1nc(Br)cnc1N)=O)C2 87808,Nc1ccc(C(=O)NCC2CCCC2NC(C2COCCN2C)=O)nc1 87809,C1(CNC(C(CC2(C(=O)OCC)CC2)=O)=O)CN(C)CCN1C.c1csc(Cl)c1 87810,N1(C(COCCC#C)=O)CC(CNC(C2CCCCN2C)=O)C(O)C1 87811,c1(C(=O)NC2CCN(C(CCC(=C)C)=O)C2)cn2ccccc2n1 87812,c1(OC)cc(OC)[nH]c(=NC2CCC(C)N(C(c3ccc4cncn4c3)=O)C2)n1 87813,c1(C(NC(=NCC2CN(C)CCO2)NC2CCC2)C)ccc2c(c1)CCCC2 87814,c1(C(N2C(C(C)NC(=O)C(F)=C3CCC3)CCC2)=O)cccc(O)c1F 87815,C=Cn1nccc1C(=O)NCC(C)CN(C)C(C1CCN(C2CC2)C1=O)=O 87816,CCCCCCCCC(=O)NCc1n[nH]cc1C(N1CCC2CCC12)=O 87817,c1(OC)ncc(S(=O)(=O)N(C(c2ccccc2Cl)CO)C)cc1C 87818,c1(NC(c2cc(Br)cnc2OC)c2n(C(CC)C)nnn2)cccc2c1OCC2 87819,C1(C(N2CC(CC)N(C(c3ccc(C)n3C)=O)CC2)=O)CN2CC3CC2(CO1)C3 87820,N1(C(C(C)=CC)=O)CCC(CNC(c2ccc(Cl)c(COC)c2)=O)C12CC2 87821,Cc1csc2ncnc(N3CCCC(CC(=O)Nc4cnnn4C)C3)c12 87822,c1(CC(=O)NC(C)CCNC(c2csc(-c3cnc[nH]3)n2)=O)c[nH]c(=N)nc1O 87823,C12(CNC(C=Cc3ccc(C)nc3)=O)CCCC1N(C(c1sccc1C)=O)CC2 87824,C(CC(F)F)(C(=O)N(C(C)C(=O)NC)C)N(C(CCN(C)CC)=O)C 87825,C=CCC(C(=O)NCC(F)C1CCC1)NC(=O)CCCN(C)C 87826,Cc1nc(NCc2nnc(-c3ccsc3)s2)cc(=NCc2ccc(F)cc2Br)[nH]1 87827,C1(CCNC(C=C(C)CNC(=O)C=CCO)=O)CCCCC1C 87828,c1(C2C(C(=O)NCCOCCNC(=O)CC3CC=CC3)C2)nc(S)n[nH]1 87829,c1(NC(C)=O)ccc(C(N2CCCC(NC(C3CCCS3)=O)C2)=O)c(Cl)c1 87830,c1(C(N2C(C(=O)NCC3(CC)CCCC3)C=CC2)=O)coc2c1COC2 87831,N1(C(CC(C)C)=O)CC2CCN(Cc3ccc4ncsc4c3)CC2C1 87832,c1(-n2cc(C3N(C(c4cnn(CC)c4Cl)=O)CCC3C)nn2)cc(F)cc(Cl)c1 87833,c1(OCC(N2C(C3(NC(c4c(CC)non4)=O)CC3)CCC2)=O)ccc(C#N)cc1 87834,c1(CC)nn(C)c(CC)c1CC(=O)NCC(C)(C)NC(c1cc(N)cnc1C)=O 87835,N1(CC(=O)N(C(CNC(C(CC)C#N)=O)C)C)C(=O)NC2(CCCCC2)C1=O 87836,C(c1c(C)nn(C)c1Cl)=CC(=O)NCC(CC)NC(C1CN2CCCN1CC2)=O 87837,C1(C(N(CCC)CCNC(C2CC=CCC2)=O)=O)CCN(C(=O)OCC)CC1 87838,N1(C(C2N(C(CCC(C)NC(C)=O)=O)CCC2CC)=O)CCC2(CC1)CN(C)C2 87839,c1(C(=O)NC(C(C)C)C(C)NC(=O)Cc2cncs2)cccc2c1OCC2(C)C 87840,CC1CCN(C(C2CCC=CO2)C(=O)Nc2ccc(Cl)cc2F)CCS1 87841,FC1(F)CCCC(c2nc(-c3ncccc3Br)no2)CC1 87842,C(=O)(C1CCCc2ccccc21)NC(CN=c1[nH]nc(C(=O)OC)s1)C 87843,CCC(C)C(O)CC(=O)N1CCC(CC(=O)NCC=C(Cl)Cl)CC1 87844,C(CO)(CCCNC(c1ccc(=N)[nH]c1)=O)NC(c1c(CC)cco1)=O 87845,c1(OCC(=O)N(C2CCN(C(C3(CC)CC3)=O)C2)CCO)ccccc1[N+](=O)[O-] 87846,C1(NC(CCc2cnc(C)o2)=O)CCCC(C(=O)N(CC(C)O)CC(C)O)CC1 87847,Cc1cnn(C)c1CC(=O)NCC1(CNC(C2CC2C)=O)CCCC1 87848,CCC(C)(C(=O)O)n1nnc(C(C)OC2CC(n3cc(CO)nn3)C2)n1 87849,c1(CNC(c2cnn(C)n2)=O)ncc(C(=O)N(C)CCOCC2CC2)cn1 87850,C(CNC(=O)C(C)Oc1ccc(F)cc1)(CC(C)C)NC(c1c(CC)ocn1)=O 87851,c1(NC(C2(CC)CN(C(=O)Cc3ccoc3C)C2)=O)cnccc1CO 87852,C(C)(CCCCNC(=O)C(F)CC1CCOC1)NC(c1ccc(C)o1)=O 87853,C1(C(N2C(C(N(CCO)CC)=O)CC2)=O)CCCSC1 87854,Cc1cc(C)c(C(=O)NCC(C)(C(C)C)NC(C2CCNC2=O)=O)o1 87855,C1(C(=O)NCC(C(=O)Nc2cn(CC(N)=O)nc2)O)CC=CC(O)C1 87856,c1(OCC(=O)NCC23CC(NC(=O)CC4C=CCC4)(CO2)C3)cccc(Cl)c1 87857,CC1(C(=O)NC2CCC(NC(=O)CCOC3CCCC3)C2)CCc2ccccc21 87858,N1(C(COC(C)=O)=O)CC2C3CCC(C2C1)N(C(=O)CC1CCC2CC12)C3 87859,N1(C(c2c(CC)nccc2)=O)CCC2(CCCN2C(C23CCC2CC3)=O)C1 87860,N1(C(c2c(C)c[nH]n2)=O)CCC(CN(C(=O)COC2CCCCC2C)C)CC1 87861,CC1(C)CC(NC(c2coc(C3CC3)n2)=O)CN(C(=O)Cc2n[nH]c(=N)s2)C1 87862,C1(C(=O)NCCCOCC2CCC2)CN(C(C2CCCSC2)=O)CC12CC2 87863,c1(NC)ccc2cc(C(N3CCN(CCOC)C(C)C3)=O)ccc2n1 87864,C1(CC(=O)N(CCNC(=O)CCn2cncn2)CC)CC(C2CC2)C1 87865,Cc1ccc(C#N)cc1C(=O)NCc1ncoc1CCNC(C1CCC1C)=O 87866,CC#CCC(C(=O)N1CCCC(CC)(CO)C1)NC(=O)C=CCOC 87867,c1(SCCOCCNC(CCNC(CN(CCC#C)C)=O)=O)ccc(O)cc1F 87868,C(=O)(CS(=O)(=O)CCOC)NC(C1N(C(C(C(CC)C)OC)=O)CCC1)C 87869,c1(C(=O)NCC2C3CN(C(=O)CC4C=CCCC4)CC23)cc(F)cc(F)c1 87870,C1(C(=O)NCC(O)CO)(OC)CCN(Cc2ccc(F)cc2)CC1 87871,C1(CCC)CN(C(C2CCCSC2)=O)CCN1C(=O)CC1CCC1 87872,c1(C(N2C(CCNC(c3c(CC)nn(C)c3)=O)COCC2)=O)ccc(F)cc1Cl 87873,C1(NC(C(CC#C)C2CC2)=O)CC2CC1N(C(=O)C=Cc1ccccc1)C2 87874,C(=O)(C(CCSC)OC)N(C1CCN(C(=O)Cc2ccn(C)c2)C1)CCOC 87875,c1(NC(C2CN(Cc3ccc(OC)cc3C#N)C2)=O)cccc2c1OCC(=O)N2 87876,C1(C(N2CC(NC(=O)OC)C2)=O)CCC(O)CN1C(=O)CC1CCN(C)CC1 87877,N1(C(CS(CC)(=O)=O)=O)CCCN(C(C2CC(F)C2)=O)C(CO)C1 87878,C(=O)(C(C)(C)S(=O)(=O)C1CC1)NC(CC1CN(C(c2c(C)cccc2Cl)=O)C1)C 87879,c1(C(C(=O)NCCc2cccc(C#C)c2)C)ccc2c(c1)OCO2 87880,N1(C(=O)NCC=C(CCC)C)CCC(C)(C(=O)OC(C)=O)CC1 87881,N1(C(CC(C(=O)OC)C)=O)CCC(C)(C)CC1C(=O)NCC(CO)OC 87882,c1(NC(c2c(OCC#C)cccn2)=O)ccc(Br)cc1Sc1cc(C)cc(C)c1 87883,C12COCCN(C1)C(=O)C2.C(C(=O)NCCSCCOC)=CCC 87884,c1(SC)cccc(C(N2CCC(C)C2CNC(=O)C2=CCSC2)=O)n1 87885,c1(-c2nc(CCNC(=O)NCC3(CO)CCOCC3)sc2)cccc(F)c1 87886,Cn1c(NC(=O)C(c2ccccc2Cl)F)nnc1C1CCCC1 87887,C(C)(C)(CC(F)C(=O)NC1(C)CC2CCC1C2)NC(C(CCCC)O)=O 87888,CC1(C)CC(CNC(C2OCC3CCCC23)=O)CN1C(c1cnc(Cl)c(N)c1)=O 87889,C1(C(=O)NC2(C)CN(C(=O)CC3(O)CCOC3)C2)Cc2c(F)cccc2O1 87890,N1(C(c2c(C)c[nH]c2)=O)CCN(C(=O)CCc2cncnc2)CC(C)C1 87891,C1(CN(C2(CN)CCC2)C(C)C)CCCOC1c1cn[nH]c1.C1C=CCC1 87892,C=CC1(O)CCN(C(=O)CC(COC)NC(c2cncc(CC)c2)=O)C1 87893,C(=O)(C(C1=CCCCCCC1)N(C)CC1CC(O)C1)NC(CC)(C)C 87894,CCCCCCCCCCCC(=O)N1CCCC1CN(C)Cc1nnc(CC)o1 87895,C(C(C)(C)CC1COC1)OC(C)=O.C(=O)(C(C)(C)C)N1C2C(C2)C1=O 87896,c1(OC)cccc(C(=O)N(C2CCCN(C(c3cnc(C)o3)=O)C2)CCF)n1 87897,C(C(CC(=O)NCCOC(=N)O)NC(C1C=CCS1)=O)OC 87898,c1(NC(CCC)=O)cncc(CCC(N2CCN(CCC#N)CC2)=O)n1 87899,c1(CCCC)ccc(CC(=O)N(C2CCC(SC)C2)C)cc1 87900,C1(C(=O)NCCC(=O)OCC)CC12CCN(c1nccc(Br)n1)CC2 87901,CC(C(=O)Nc1cnc(F)nc1)C(C)NC(c1ncc(F)cn1)=O 87902,CCCC(C)(C)C(=O)NCC(CNC(c1cnn(C)c(=O)c1)=O)OC 87903,CC1C(NC(C2CCN(CC3CC3)CC2)=O)CCCN1C(C12CC1CNC2=O)=O 87904,N1(C(C(c2ccc(C)cc2)F)=O)CCC2C(CCCN2C(C2CCS2(=O)=O)=O)C1 87905,N1(C(COC(CC)C)=O)CCC2CCN(C(=O)Cc3nc(C)sc3Cl)C2C1 87906,N1(C(C(C)Oc2ccc(C)cc2C)=O)CCN(C(=O)CSC(F)F)CC(O)C1 87907,CC(C)C(CNC(C1(C)CC1(C)C)=O)C(=O)NCc1c(F)cccc1F 87908,c1(C(C)=O)ccc(CC(N2CC=CC(NC(=O)CCN3CCC(F)C3)C2)=O)cc1 87909,c1(CCC(=O)NC2C(CNC(CC)=O)C2)cccc(CC#N)c1 87910,C1(CNC(C(C)OC(F)F)=O)CC(C)CN(C(=O)CN2C(=O)CNC2=O)C1 87911,C1(C(=O)OCC)CN(C(=O)CC2CCC(O)C2O)CC1(C)C 87912,C(N=c1[nH]c(=NCC(C(C)C)N(C)C)[nH]c2c1CCCCC2)c1snc(C)n1 87913,CC1(CCCCNC(=O)COC2CN(C(=O)CCN=[N+]=[N-])C2)CC1(F)Cl 87914,c1(C(=O)NC2CCN(C(C3CC4C(C3)C4(F)F)=O)CC2F)occ2c1CCOC2 87915,C(c1cccc(C#N)c1)=CC(=O)NC1C(OC)CN(C(C2CCCO2)=O)C1 87916,N1(C(C2(C)C(C)(C)C2)=O)CC2COCC(C1)C2NC(=O)C1=C(Cl)CC1 87917,N1(C(C(CC)OCC)=O)CCCC2CN(Cc3ccc(S(C)(=O)=O)cc3)CCC12 87918,c1(CC(N2CCCC(N(C(=O)C(C#N)C(C)C)CC)C2)=O)nc2ncccn2n1 87919,c1(CNC(=O)CC(C)NC(C2(C(=O)OC)CC2)=O)cccc(F)c1F 87920,C1(NC(=O)CCc2nnc(C(F)F)o2)CCCC1C(=O)O 87921,c1(C(N(C2CCN(C(c3[nH]ccc3COCC)=O)C2)C)=O)cccnc1S 87922,CCC(C)(O)C(=O)NCC1CC(OC)CN1C(=O)CCc1ccco1 87923,N1(C(C(C)OC(C)(C)C)=O)CCC2(CCOCC2)C(NC(=O)C=CCO)C1 87924,C1(CC)CCN(C(=O)C=Cc2ccnn2CC)C1C(=O)NCc1cnn(C)c1 87925,N1(C(CN(CCOC)C)=O)CCC(NC(=O)C(C)(C)NN2CCCC2)C(C)C1 87926,C(CCCCCC(=O)NC(C1CCN(C(c2ccc(C(N)=O)cc2)=O)C1)C)SC 87927,N1(C(c2cn(C)nc2O)=O)CC(CO)C2(C1)CN(C(=O)C(C)(C)n1cncn1)C2 87928,Cc1ccc(C=CC(=O)NC(C)CN(C(=O)CC23CCCC2C3)C)cc1 87929,CCS(=O)(=O)CC(=O)N1C2CCC(C2)C1C(=O)NC(CO)C1(C)CC1 87930,C(CC(C)(C)C)(C(=O)N1CCC(C)(C(N2CCCCC2)=O)C1)OC 87931,C12(C(=O)NCC3C=CC(NC(=O)Cn4cc(Cl)cn4)C3)CCC(F)(CC1)CC2 87932,c1(C(N2CC(CN(C)Cc3ccc(Br)c(F)c3F)C2)=O)cc2cccnn2n1 87933,C(CCCCC(=O)NCC1CCC(C#N)C1)n1cc(C2(CC)CCC2)nn1 87934,N1(C(c2c(Cl)cc(C)s2)=O)CCC2(CC1)CC2NC(=O)CCC1CCCN(C)C1 87935,N1(C(c2c(OC)nsc2)=O)C2CCC1C(C)C(NC(=O)CC(C)C1CC1)C2 87936,C1(CNC(c2c(C)nn(C)c2Cl)=O)CC(N=c2ccnc(S(C)(=O)=O)[nH]2)C1 87937,c1(C(=O)NC2CCC(C)N(C(=O)Cn3ncccc3=O)C2)ccn2c1CSCC2 87938,C1(NC(C(=Cc2cccnc2)C)=O)CCN(C(=O)CC2(C)CCC2)CCC1CO 87939,CC1CN(Cc2cc(-c3cc[nH]c(=N)c3)ccc2F)C(C)(C)C1 87940,C(=O)(N=c1ccn(CCF)[nH]1)C1(C=C)CCN(C(=O)CCC2CCCOC2)C1 87941,c1(NC(C(n2cc(CCOC)nn2)C)=O)ccccc1[N+](=O)[O-] 87942,C(c1ccccc1)=CC(=O)NCC1C(CC(N2CC(OCC(=O)N(C)C)C2)=O)C1 87943,c1(C(N(CCNC(=O)C(F)OC)CC)=O)n[nH]c(C(C)C)c1[N+](=O)[O-] 87944,C(=O)(C1=C(C#N)CCC1)N1CC(NC(c2c(CCC)n(C)nn2)=O)C(SC)C1 87945,N1(c2nnc(C(C)(C)C)s2)Cc2nccn2CC(NC(C2(C)CC2(F)Cl)=O)C1 87946,C=CCC(C)(CC)C(=O)NC1CCCC1CNC(c1cnnn1C)=O 87947,c1(OCC)nc(C)ccc1CNC(C1CCCN1C(=O)CCC(C)C#N)=O 87948,c1(C(N2CCC(N(C(c3cc(C)on3)=O)C)C2)=O)c(-n2nccn2)cccc1F 87949,C1(C(=O)O)(C(=O)NCc2ccccc2)CN(C(C2CCCC2)C2CCC2)C1 87950,Cc1nc(C(C)C)ccc1C(=O)NC1CCCC(NC(c2cc(F)n(C)n2)=O)C1 87951,C(=O)(C(C)(C)C(=O)NC1CCCC(C(=O)NCC2CCCCC2)CC1)OCC 87952,c1(C(C(=O)OCC)C(=O)NC2CCCOC2)ccccc1F 87953,C1(CCC)CN(C(=O)CCNC(=O)COC)CCN1C(C1CCCOCC1)=O 87954,C(=O)(CS(=O)(=O)C1CCCC1)NCC(C(C)(C)C)NC(C1CC2(C1)CC2(F)F)=O 87955,Cc1ccc2snc(C(=O)N(CC(C)NC(C3CC4CCCCN4C3)=O)C)c2c1 87956,C1(NC(Cc2ccn(C(C)C)n2)=O)COC2(C1)CN(C(C1CCCOCC1)=O)C2 87957,CC1OCCCC1C(=O)NC1(C(=O)NCC(C)(O)C2(C)CC2)CCCCC1 87958,Cc1ncnc(C)c1C(=O)NCCCC(c1ccccc1)Nc1ccc(C#N)nc1 87959,CCC(C(=O)NC1CC(CNC(=O)C=Cc2cc[nH]n2)C1)n1ccnc1 87960,C(CN=C(NCC1CC=CCC1)NC(C)CC(F)F)OCC 87961,Cc1cccc([N+](=O)[O-])c1C(=O)NCC(n1cc(CCCO)nn1)C 87962,N1(C(=O)NC)CCCC(CCC(N2CCC(C(C)O)CC2)=O)C1.C1(C)CC(=O)O1 87963,O(NC(=O)C(F)C(C)CNC(c1ccc(C)c(C)c1)=O)CCCC#C 87964,CC1(NC(=O)CC2CCSCC2)CCCN(C(c2coc(CC3CC3)n2)=O)C1 87965,C1(O)(C(c2ccsc2)NC(c2cc(OC)no2)=O)CCN(C(=O)CCC2CCC2)C1 87966,C1(CCC(=O)NCC2CC2C)(NC(CNC(=O)OCC)=O)CCC1 87967,N1(C(c2ncn3c2CCC3)=O)CCC2(CCSCC2)C1 87968,CC1CN(C(c2occ3c2CCC3)=O)CCCN1C(C1CCC2(CCC2)C1)=O 87969,C1(CC(=O)NCC(C)NC(C(COC)C)=O)(CNC(C)=O)CCCCC1 87970,c12cc(C)c(c(C)c1)CC=CC(=O)N2.c1(C(=O)OCC)onc(C(=O)O)c1C 87971,C1(C(N(CCNC(=O)Cc2csc(S)n2)Cc2ccccc2)=O)CCCC1(F)F 87972,N1(C(C(CCSC)OC)=O)CC2CC1CN2C(c1ncn(C(C)(C)C)n1)=O 87973,Cc1cc(Cl)ncc1NC(N1CCOCC1c1noc(C(C)C)n1)=O 87974,C1(CC)CCC(O)(C(=O)NCCC2(CNC(=O)C=Cc3ccc[nH]3)CC2)C1 87975,C#Cc1cc(F)c(C(=O)NC(CO)C(C)NC(c2cnnn2C2CC2)=O)cc1F 87976,C12(c3ccn(C)n3)CCC(C1)C2C(N1CCC1CNC(C1(CF)CC1)=O)=O 87977,C(CCC(=O)N1CCCC1C(C)NC(=O)C(C)N1CC(C)C1)OCC 87978,CP(C)(=O)C(O)C(=O)N1CCC(NC(c2cnc[nH]2)=O)C(O)C1 87979,c1(C(=O)NC(C)CCNC(C2(CCF)CC2)=O)cc([N+](=O)[O-])ccc1OC(F)F 87980,c1(C(c2nnnn2Cc2ccco2)NCCC(C)O)cc(F)cc(C#N)c1 87981,c1(OCCN(CCOC)C(=O)Nc2cnsc2)ccc(Cl)c(C)c1 87982,Cc1cc(C(=O)N(C)CC2CCN(C(=O)C=Cc3cn[nH]c3)C2)no1 87983,CC(C(F)F)N(C)N(C)CCc1c[nH]c2ccccc12 87984,c1(C(=O)NCC(CC)NC(CSCC#C)=O)cn(C)nc1OC 87985,Cc1cncc(C)c1C(=O)NC(CCN(C)C(c1cc(C(N)=O)c[nH]1)=O)C(C)C 87986,N1(C(c2c(CN=[N+]=[N-])ccs2)=O)CCN(C2CCN(C(C3(CF)CC3)=O)C2)CC1 87987,c1(CC(N2C(C)C(C(=O)NCC3(CO)CC(C)(C)C3)CC2)=O)ncc(F)cc1F 87988,Cc1nc(C(N2CC(O)C(O)C2CNC(=O)CCCc2nccs2)=O)cc(O)n1 87989,CC1=C(C(=O)N2CC=CC(NC(C3CCCSC3)=O)C2)CCCO1 87990,c1(N(CCCS(C)(=O)=O)C)nc(-c2ccccc2)nc(=NC2CCOC2C)[nH]1 87991,C1(C(N(CCOC)CCO)=O)CCC2(CC2)N1C(C1Cc2nccn2C1)=O 87992,N1(C(Cc2cccc(C#C)c2)=O)CCC2(CCCN(C(=O)CCCOC)C2)C1 87993,N1(C(c2ccc(C)cn2)=O)CC2(CCOCC2)CC1CNC(=O)C(C)C1CC1 87994,C1(C(=O)NCC(CNC(c2c(C(C)C)sc(Cl)n2)=O)F)Cc2cccnc2C1 87995,C1(NC(C(C=CCCC)O)=O)CCCC(NC(C2CC(=O)N(C(C)(C)C)C2)=O)C1 87996,c1(C(N(CCC(C)NC(=O)CN2CCOCC2)C)=O)cc2c(F)c(F)ccc2s1 87997,c1(C(N2CC(CNC(c3cn(C)[nH]c3=N)=O)OCCC2)=O)cccc2cncn12 87998,C1(CNC(CNC(CNC(CC=CC)=O)=O)=O)CCCC(C#C)C1 87999,c1(OCC(=O)N(CCN(C(C2CCC2(C)C)=O)CC)CC)ccc(C#N)cc1 88000,C1(CC(C(=O)NC(CC)C)N(C(C)C)Cc2cc(C)n(C)n2)CCN(C)CC1 88001,c1(C(=O)NCC2N(C(C3C(C(C)(F)F)C3)=O)CC3(CC3)C2)ncc2[nH]ncc2n1 88002,c1(C(N2CCC(C)(NC(C3CCC4CC4C3)=O)C2)=O)cc2n(n1)CCNC2=O 88003,C(=O)(C(F)CCC(C)C)NCC(CC(F)(F)F)NC(C(C)SCC)=O 88004,C1(c2nn[nH]n2)(C(=O)NC(C(C)C)c2nc[nH]n2)CC12CCCC2 88005,c1(C(=O)NCCOCCNC(c2c(C)nncc2)=O)cccc(CO)c1C 88006,c1(OC)cc(S(=O)(=O)N2CC(CNC(c3cc4cccnc4[nH]3)=O)C2)ccc1Br 88007,n1(CC(=O)NCC2CC(NC(C3CCC(=O)O3)=O)C2)c(=O)cnc2ccccc12 88008,c1(C(=O)NC(C2CCCC2)CNC(c2n(CC#C)ccc2)=O)ncccc1CO 88009,C=CC1(C(=O)NCC(c2ccc(F)cc2)NC(C2CC2C)=O)CCOCC1 88010,C1(C)(C(N(CC=C)C)=O)CCN(CC2(N(C)C)CC2)CC1 88011,CC1CCCC(n2nc(-c3ccc(N(C)C)nc3)nc2CCF)C1 88012,c1(C(C(=O)NC(C(=O)NCC(=C)Br)C2CC2)C)cncnc1 88013,N1(C(C(CCC)N(C)C)=O)CCC2(CC1)CN(C(=O)Cc1ccc(CC)cc1)C2 88014,N1(C(C2C(=C)C2)=O)CCCCC12CC(NC(=O)CCCSCc1ccccc1)C2 88015,C1(CNC(c2c(C)cc[nH]2)=O)CC2CCC(C1)N2C(=O)Cc1nonc1C 88016,CCC(CC)C(C)C(=O)NCC1(OC)CN(C(=O)COCC(C)C)C1 88017,Cn1cnc2nc(N3CCN4C(=O)N(C)CC4C3)nc(NCC3(C)CC3(F)F)c12 88018,CN1CCC(NC(=O)OC2CCCCC2)C1c1cccs1 88019,N1(C(c2nccc(OC)c2)=O)CCCC(O)(CNC(C2CC3(CCC3)CO2)=O)C1 88020,C12(C(=O)NCCCOCCN(C)C(C3CC(F)(F)CS3)=O)CCC(CC1)CC2 88021,n1(CC(=O)NC(CC)CN(C(=O)CCSc2nccn2C)C)cnc([N+](=O)[O-])c1 88022,CC1CC(NC(=O)Nc2ncccn2)c2nccn21 88023,c1(C(=O)NC(C)CCNC(c2nnn(C(C)(C)C)n2)=O)cc(Cl)ccc1[N+](=O)[O-] 88024,C(=O)(C(CO)C(F)(F)F)NC1C2C(C(=O)NC(C(=O)NC)CC3CC3)C3C(C2)C13 88025,C1(c2ccc(CC)o2)NC(=O)N(C2CC2)C2=C1C(=O)N(C1CC1)CC2 88026,C1(CCCC)CN(C(=O)Nc2cc(C(C)(F)F)ccc2Cl)CCN1CCOC 88027,c12cc(Cl)ccc1OC2.C(=O)(C(C)N(CCNC(C)=O)C1CC1)OC 88028,c1(NCCn2c(-c3n(CC=C)nnn3)c(C)cn2)ccc(OC2CCOC2)cc1 88029,c1(C(=O)NC(C2(O)CN(C(=O)C=CC3(C)CCC3)C2)C)ncoc1C1CCC1 88030,c1(CNC(CCN(C)CC)=O)cn(CC(=O)N(CCC(C)(C)O)C)nn1 88031,Cc1c(NCC2CCCC(F)(F)C2)ncnc1N1CC(C)SC(C)C1 88032,C1(C(C)C)CCOC1C(=O)N(C)CC1(O)CN(C(=O)C(C)CN2CCCCC2)C1 88033,c1(C(=O)NCC2(COC)CN(C(=O)CC(C)(C)C)C2)cc(F)ncc1OC 88034,C1(C)(CNC(C(C(C)C)OCC)=O)CCN(C(=O)CCc2ccoc2)CC1 88035,Cc1nc(CCC(=O)NCC2C(C)CCN2c2nnc(C3CC3)o2)[nH]c1C 88036,CCCCC(C)CCC(=O)NC1CCCC1(C)CNC(=O)CNC(=O)CC(C)C 88037,C1(C(N(C)CCNC(=O)Cc2cncnc2)=O)CCNC(=O)C1 88038,N1(C(C(=O)NCC=C)C)CCC(O)(C(=O)NCC(C2CCCCC2)C)CC1 88039,c1(CNC(C2(F)CCN(C(c3cncc(Cl)c3)=O)C2)=O)ccnc(F)c1F 88040,Cc1ccc(Br)c(NC(C2CC(NC(=O)Cn3cc(Cl)cn3)C2)=O)c1 88041,C1(C#N)(C(N(C(CNC(c2ccsc2)=O)Cc2ccccc2)C)=O)CCOCC1 88042,CON=CC(=O)NCCCCC1CN(C(c2csc(CC(F)(F)F)n2)=O)C1 88043,C1(C(=O)NC(C(=O)OC)C2CC2)CSCCN1C(c1cnc(O)[nH]1)=O 88044,n1(CCC)ncc(-c2nc(C3CCCCCC3)nn2C(C)C(C)C)c1C 88045,Cc1[nH]c(C)c(C(=O)N(C)CCOCCN(C)C(C2(C)CCN(C)C2)=O)c1C 88046,C1(CNC(Cc2cc(C)ns2)=O)CCCCN(C(=O)C(N2CCSCC2)C)C1 88047,CC#CCCCC(=O)N1CCCC(CCNC(=O)C(C)CSC(F)(F)F)CC1 88048,CC(C)(C)CCCC(=O)N1C(CNC(C2(C)CCNC(=O)C2)=O)CC2COCC12 88049,N1(C(c2cc(Br)ncc2F)C(=O)NC(C)C)CC(C)C2CCCCC12 88050,N1(C(C=CCCC)=O)CCC(C(C)(C)NC(=O)CCn2cc(C)cn2)CC1 88051,C1(F)(C(=O)NC(C2CCOC2)CC)CCN(C(c2ccn(COC)n2)=O)CC1 88052,N1(C(C(=O)Nc2c(OC)cc(Cl)c(C)c2)=O)CCC(C2CCC(F)(F)CC2)C1 88053,N1(C(CCSCCC)=O)CC2(CCCN(C(=O)C(C)(O)Cc3ccccc3)C2)C1 88054,C(=O)(C1=C2CCCN=C2NN1)NC(C1CCCN(C(CCC=CCC=C)=O)C1)C 88055,C1(CC(=O)NCCOCCN(C)C(c2cc(C#N)on2)=O)SC2=NCCN2C1=O 88056,C(=O)(CCCC(F)(F)F)NC(CSCC)C(=O)NCCC1CCN(C)C1 88057,C1(NC(c2ccc(CNC(c3ccc(C#C)o3)=O)s2)=O)CCC(C)(C)CC1 88058,c1(C(C(=O)NCC(CNC(c2c(OC)n(C)nc2)=O)CO)=O)cc(F)ccc1C 88059,N1(C(CCC#C)=O)CCC2CC2(NC(=O)CCNC(c2ccc(F)cc2)=O)CC1 88060,CN1CC(CC(=O)N(C)CCc2cn(-c3ccc(I)cc3)nn2)C(O)C1 88061,N1(C(c2nnn(CC)c2C)=O)CC(C)N(C(c2cccc(COC)c2)=O)CC1C 88062,C(=O)(C(C)(C)C(F)F)NC1CC(NC(c2ccn(CCOCCOC)n2)=O)C1 88063,O=C(C1=CCCC1)NCC1(O)CC(C(N2CC(N3CC(O)C3)C2)=O)C1 88064,C1(CNC(c2n(C(C)C)nnc2)=O)CN(C(=O)CNc2ccccn2)CC12CC2 88065,N1(C(C2C(C)=C2)=O)CC2CCN(C(=O)C(F)(F)C3CCCC3)CCC2C1 88066,c1(OC)c(C(N2C3CCC2CC(NC(c2ccnn2C)=O)C3)=O)ccc(Cl)c1C 88067,C1(C(=O)NC2C(CC(=O)NC(C#C)CCC)C(O)C2)NC(=O)OC1C 88068,C1(CC(=O)NCC#C)CCN(C(C(CC)CC)=O)CC1 88069,C#CC1(C(=O)NCCCCc2nc(-c3ccccc3)no2)CNC1 88070,Cc1nc2ccc(C(=O)NC3CC3CNC(C3(C)COC(=O)OC3)=O)cc2o1 88071,C12(C(=O)NC3C(CN(C)C(c4ccc(C(N)=O)nc4)=O)CCC3)CCC(CC1)C2 88072,C(=O)(C(C)(C)CCS(C)(=O)=O)NC(Cc1ccc(OC)cc1)(C)C 88073,N1(C(CNS(CC)(=O)=O)=O)CC2CC(C1)C(CO)C2NC(=O)C(C)(CC)OC 88074,CC1(C)CCCCC(C(=O)NCC2CN(C(c3ncccn3)=O)C2)C1 88075,CC1CN(C(=O)CCc2cnc(O)[nH]2)CC1n1cc(CC2CC3CCCC23)nn1 88076,C1(C(=O)NC(c2cn(C)nn2)C(=O)NCc2c(OC)n(C)nc2)CCC(C2CC2)C1 88077,C12(C(N(C(C=C)C)C)=O)CC1CN(C(=O)C=Cc1ccoc1)C2 88078,N1(C(Cc2cc(C)no2)=O)CC2CCCC(NC(C3CCCOCC3)=O)(C2)C1 88079,C1(CC)CCCC1(C)C(=O)NCC1CCN(C(=O)Cc2cccc(OCC)c2)C1 88080,C1(OCC#C)CCCN(C(=O)CONC(=O)Cc2cccnc2)C1 88081,c1(C(N2CCC(C(C)NC(C3CCN(C)C3)=O)C2)=O)ccc(F)nc1 88082,Cc1ncc(C(N2CCC(C)C(CNC(c3ccc(O)cc3O)=O)C2)=O)c(C)n1 88083,c1(C(N(CCNC(c2cc(S(=O)(=O)NC)oc2)=O)C)=O)ccc2sc(C)nc2c1 88084,n1(CCC(=O)NC2CN(C(C3CC34CC4)=O)CC2O)ncc(=O)c2ccccc12 88085,Cc1ncnc(C)c1OCC(N1CCN(C(C2CC2F)=O)C(C(C)C)C1)=O 88086,c1(CC)cnc(C(N2CCC(NC(=O)C(C3CCCO3)C3CC3)C2C)=O)cn1 88087,C=CCC(C(=O)NCc1nccn1C)NC(C1CCCC1CCC)=O 88088,c1(CC(=O)NC)cccc(C(=O)NCC2C3CN(C(C)C=C(C)C)CC23)c1 88089,c1(C(=O)NCC(CNC(c2c(C)onc2)=O)(C)C)nn2c(c1Br)CCC2 88090,CCCC(CC(=O)Nc1cscc1C)NC(C1CCCN(C)C1)=O 88091,c1(C(N2CCC(OCC)C2)=O)cc(CN(C)C)nc(Cl)c1.C1CCCC(=O)N1 88092,C1(NC(CSCC)=O)CCCC(N(C(=O)CC2CN(C)C2)C)C1 88093,C(C(O)C(=O)NCC(C)N(C(=O)CNC(=O)NC)C)=CCCC 88094,c1(C(=O)NCCCCC(C)NC(CSCCCC)=O)cccc2c1OCCN2C 88095,Cc1ncnc(C(N2CCSCC2C(=O)N(CCCCC(C)C)C)=O)c1C 88096,Cc1cc(-c2ccsc2)ncc1C(=O)NC1CCC(NC(c2cscn2)=O)CC1 88097,N1(C(CN2CCN(C(CC3N(C)CC=CC3)=O)CC2)=O)CC(=O)NCC12CC2 88098,N1(C(c2n(C)ncn2)=O)CC2C(NC(c3cccc(Br)c3)=O)C2C1 88099,c1(OC)ccc2c(c1)CCC2C(=O)NC(CNC(C12CC(F)(C1)C2)=O)CC(C)C 88100,C1(NC(C2CC(=C)C2)=O)CCCN(C(c2ccc(C#N)c(O)c2)=O)CC1F 88101,Cc1cc(NC(=O)CS(=O)(=O)C2CC2)ccc1S(C)(=O)=O.C1CO1 88102,c1(CC(C)NCc2cccc(P(C)(C)=O)c2)ccc2c(c1)CC(C)O2 88103,C1(NC(c2ncc(C)nc2)=O)CC2CC1CC2C(=O)N(C1CC1C)C 88104,Cc1nc(C)n(CC(=O)NCC(O)CCNC(C2CCN(C3CC3)C2=O)=O)n1 88105,C1(C(C)C)N(C(c2cnc3c[nH]nc3c2)=O)CC12CCN(C(=O)C1CC1)CC2 88106,c1(CCC(=O)NCCC(C)CCNC(C2(F)CCCCC2)=O)cccc(Cl)c1Cl 88107,N1(C(C=CSC)=O)CCCC(C)(C)C1CNC(C1C2CCCOC12)=O 88108,CC(C)CCC(C(=O)NC1CCS(=O)(=O)C1)NC(C1CCCC(=O)N1C)=O 88109,CC(CCCNC(c1cnc[nH]1)=O)NC(=O)CCc1nccn1C 88110,C1(CCC)CCN(C(C2CC(CCNC(=O)C(F)OC(F)(F)F)C2)=O)C1 88111,C1(C(=O)NCC(CNC(C(Cn2ccc(C)n2)C)=O)O)CC(C2CC2)=NO1 88112,C1(OC)CC(NC(C2(OC)CCSC2)=O)CN(C(=O)Cc2occc2C)C1 88113,c1(CNC(CCC(C)N(C)C)=O)cccc2nccnc12 88114,CC(C)CC(C)(O)C(=O)NCC1CCN(C(c2ccc(CN(C)C)[nH]2)=O)C1 88115,N1(C(CCCCOC)=O)CC(NC(C2(C(=O)N(C)C)CC2)=O)CC(F)(F)C1 88116,Cc1ccc(O)c(C(N2CCC(O)C(NC(C3CC4(C3)CC4F)=O)C2)=O)n1 88117,C1(C(=O)NC(COC)C2CC2)CC2(CCN1C(c1cnn(C)c1C)=O)CC2 88118,N1(C(CCC)=O)CCC2(C=C(C(=O)N(C)Cc3cncs3)C2)C1 88119,N1(C(C(C)Oc2ccccc2Cl)=O)CC(NC(=O)Cc2ccoc2)C2CC2C1 88120,C1(C(=O)NCCn2ccnc2)CN(C(c2ccnc(-c3ccccc3)c2)=O)CCN1 88121,CP(C)(=O)c1ccc(C(=O)NC2(C)CC(NC(c3n[nH]cc3Cl)=O)C2)o1 88122,c1(CC(N2CC=CC(NC(CCCCSC)=O)C2)=O)cnc2n1CCCC2C 88123,CC1(C)CCCN1CCC(=O)NCCn1cc(C(c2ccccn2)O)nn1 88124,c1(SCNC(C(c2ncc(CC)o2)N(CCC2CC2)CC)=O)ccc(Br)cc1 88125,c1(C(=O)NCC2CCN2C(C23CC(F)(C2)C3)=O)cnc2ccsc2c1 88126,C=C(C)CC(C)C(=O)NC1CN(C(c2csc(CO)n2)=O)CC1O 88127,c1(NC(=O)NC2C=CCN(C(C3CCCO3)=O)C2)ccc(Br)cn1 88128,C(c1cccc(C#N)c1)=CC(=O)NCCC(C)NC(c1c[nH]nc1C1CC1)=O 88129,c1(C(C(=O)NCc2ccsc2)N(C(C)(C)C)CC)cc(C2CC2)on1 88130,N1(C(C(C)SCCCC)=O)CCCN(C(=O)C=CSc2ccco2)C(C)C1 88131,C(=O)(C1CCCc2ncnn21)N(C)CCN(C)C(C1(C)CC2CCC1C2)=O 88132,c1(CCC(=O)NCC(CNC(c2n(CC=C)ccc2)=O)F)nc2ccccc2s1 88133,C=C(Cl)CCC(=O)N(CC(C)NC(=O)C(C)(C)c1cscc1Cl)C 88134,Cc1cccc(C(C)(C)C(=O)NCCCC(C)NC(c2nc(C(C)C)cs2)=O)c1 88135,C1(CNC(=O)C=CC2CCCC2)CN(C(C2(CC3CC3)CC2)=O)CCO1 88136,Cc1ncccc1CCCNC(C1(NC(=O)COc2ccccc2)CCCC1)=O 88137,N1(C(=O)C(O)Cc2ccccn2)CCN(C(=O)Cc2ccsn2)C(CO)C1 88138,c1(CN2CC(C(=O)Nc3cc(OC)n[nH]3)SCC2)ccc(Cl)nc1C 88139,c1(COC)ccc(C(N2CCC(N(C(=O)C(CO)NC(N)=O)C)CC2)=O)cc1 88140,c1(C(c2n(CCOCC)nnn2)NC(C2COC2)C)cccc(F)c1OC 88141,Cc1ccc(C(C)C)c(C(N2CCSC(C)(C)C2)=O)c1 88142,N1(C(CC2C(C)OC(C)C2)=O)CCN(C(c2cc3ccsc3[nH]2)=O)CC1C 88143,c1(C(N(C2CCCN(C(=O)Cc3ccccc3)CC2)C)=O)cnc2ccnn2c1 88144,C1(C)(OCC(=O)N(C)CC2(NC(CC3(CC(=O)OC)CC3)=O)CC2)CCOCC1 88145,c1(C(N2CCC(NC(C3(CC#C)CCCC3)=O)C(C)C2)=O)cc(O)cc(C#N)c1 88146,C=CC(CC)CC(=O)NN(C(C)C(=O)N(C)CCOC(C)=O)C 88147,N1(C(C(C(C)O)(C)C)=O)CC2CCC1CN2C(=O)CCc1ccccn1 88148,C1(CNC(c2ccc(C(=O)OC)o2)=O)CCCCN1C(=O)C(C1CCOCC1)F 88149,c1(CN2CC(NC(C(c3ccc(O)cc3)C)=O)C(F)(F)C2)cc(Br)cc(Br)c1O 88150,Cc1nc(O)nc(C)c1CC(N1CC(C2(NC(c3csc(C)c3N)=O)CC2)C1)=O 88151,c1(C(N2C3(c4cn(C(COC)COC)nn4)CCC2CC3)=O)ccccc1[N+](=O)[O-] 88152,N1(C(C(CNC(c2n(C)ccc2)=O)N(C)C)=O)CCOCC(C(N)=O)C1 88153,C(C)(C)(C(=O)NCC=CC(=O)NC1CC1CC(C)C)SCC 88154,c1(C(=O)NCC2C(C(=O)NCc3cn(CC)nc3)CCO2)cncc(OC)n1 88155,C(=O)(C1COc2ccccc21)N1CCC(NC(C2(CCOC)CC2)=O)C(F)C1 88156,C1(CC)(NC(=O)CCc2ccoc2)CCN(C(c2n[nH]c3c2CCC3)=O)CC1 88157,c1(NC(C(=O)NCCCOC)C)ccc(P(C)(C)=O)cc1 88158,CCCCN=C(NCCc1ccc(F)cc1F)NCC1CC(=O)N(CCC)C1 88159,CCCCC(C(=O)N(CC)CC1CCC1(F)F)C(C)C 88160,Cc1csn1CC(=O)NCCN(C(=O)CC1CCCC1)C1CC1 88161,N1(C(CCC#C)=O)CC2(CCN(C(=O)CNCCOC)C2)C1.c1(C)ccccc1 88162,C(CC(=O)NCC1CN(C(=O)C=C2CCCCC2)CC1O)(C(C)C)OCC 88163,S(=O)(=O)(c1cnn2ccc(=NC(C)CCOC)[nH]c12)NC(C(CC)CC)C 88164,C1(C(=O)NC2CC(C)(NC(c3cn(C)nc3)=O)C2)C2CCN(CC2)S1(=O)=O 88165,c1(C(N2C(CCCNC(c3cnc(S)[nH]3)=O)CCCC2)=O)ccc2nc[nH]c2n1 88166,N1(C(=O)Nc2ccnn2C2CNC2)CCC2(CCCCO2)C1 88167,C(c1ccc(F)cc1Cl)=CC(N1CC2CN(C(CCCC#C)=O)CC21)=O 88168,Cc1c(NC(c2cncc(NC(=O)Cn3ccnn3)c2)=O)ccc(Br)c1Br 88169,n1(CCC)nc(C)cc1C(=O)NC1CCC1NC(c1cccc(C(N)=O)c1)=O 88170,c1(C(=O)NCC(C2CCCC2)NC(C2N(C)CCC2)=O)ccc2nc(O)[nH]c2c1 88171,N1(C(c2cncc(NC(CC)=O)c2)=O)CCC(C)C(NC(=O)CC(C)(C)F)C1C 88172,C1(C(=O)NCC2(C)CCC2)CC(F)CN1C(=O)CN(C1CCSC1)C 88173,c1(C(N2CCC(c3cnccn3)C2)C(=O)N(C2(C)CC2)C)cnccn1 88174,Cc1ccc(F)c(C(=O)NCCC(C)(C)NC(=O)CC2CCC(O)C2)c1F 88175,CCC1=NOC(C(N2CC=CC2CNC(c2cnoc2COC)=O)=O)C1 88176,CCCCC(C(=O)NC1CCN(c2nnc(C(F)F)o2)C1C)NC(N)=O 88177,N1(C(c2n(C)ccn2)=O)CC2CCOC2(CNC(c2ccsn2)=O)C1 88178,c1(NC(Cn2cc(C(=O)OC)nn2)=O)ccc(C)c(N(C)C)c1 88179,c1(CN(c2ccccc2N2CCCCC2)CC(N2CCCCC2)=O)cc(I)ccc1O 88180,c1(OCC)ccc(NC(=O)NCCCC2(C)CC2(Cl)Cl)cc1OC 88181,c1(CC(=O)NCC2C(C(=O)NCC(N3CCOCC3)C)C2)cn(C)nn1 88182,C1(C(N(C)CC2N(C(C(C)O)=O)CCOC2)=O)CCC(C2CC2)CC1 88183,N1(CC(CC)C)CCS(=O)(=O)C(CCNC(=O)Cc2nnn(C(C)(C)C)n2)C1 88184,N1(C(CC=CC)=O)CC2CCC(C1)C2CNC(=O)C(c1ccc(C2CC2)cc1)O 88185,C1(CC(=O)Nc2ccc(O)cn2)CC(N=c2ccnc(C(F)(F)F)[nH]2)C1 88186,CC(C)CCC(O)C(=O)N(C(C)C(N1CC(O)CC(O)C1)=O)C 88187,c1(OCCNC(=NC)NCc2cnccn2)ccccc1C#N 88188,N1(C(CN(CCC)C)=O)CCC(C)(C(=O)NCC2CN(CC)CCO2)CC1 88189,C1(C)(C(=O)NC(CC2CC2)C(F)(F)F)CN(C(C2CCC(CO)CC2)=O)CC1C 88190,Cc1ccc(N)c(C(=O)NC(c2ccccc2)C(C)NC(=O)C(C)C)c1 88191,C1(N(C(=O)CCc2csc(C)n2)CC#C)CCN(C(C2CCC(C)S2)=O)CC1 88192,c1(CC(N2CC3CC(NC(CN(C)CC)=O)C3C2)=O)ccc2n[nH]cc2c1 88193,N1(C(CC(C)(C)C)=O)CC2CCCC(NC(c3coc4c(F)cccc34)=O)C2C1 88194,N1(C(CCN(C)CC)=O)CC(NC(c2cc(C(C)C)no2)=O)CC(O)C1 88195,c1(C(=O)NCC2C(NC(CCC=C)=O)CC2)c(C)ccc(F)c1O 88196,c1(C(c2nnnn2C2CCCCCC2)NCC(COCC)C)oc(CC)nc1C 88197,c1(C(N2C(CC(=O)NCCc3c(C)c[nH]c3C)COCC2)=O)nc(Cl)ccc1F 88198,C(=O)(C1CCc2c(Cl)cccc21)N(CCCNC(=O)COC1CC1)CC 88199,CC(C(=O)NC1CCCOC1C1CCN(C(C2CCCC2)=O)CC1)C(C)(F)F 88200,C(C)(C)(CCCC(=O)N1CCC2C(O)CC12)NC(CCc1n(C)cnn1)=O 88201,C(=O)(C(F)CC(C)(C)NC(c1cc2ccccn2n1)=O)N(C)CCc1cccs1 88202,C1(C(=O)NCC2C(C)CCCN2C(C2CC2C(C)O)=O)CCCC2C1C2(F)F 88203,C(C(COC)C(=O)N1CCCC(CCCO)C1)OC 88204,CCC(C)C(O)C(=O)N1CCN(C(=O)Cn2cc(C)ccc2=O)CC1 88205,c1(C(C)C)nc(C(=O)NCC(C2CCCN2C(C2CC(N(C)C)C2)=O)(C)C)cs1 88206,C(=O)(C(C)(CO)NC(C1CCCC(=O)N1)=O)N1C(C)(CC)CC1 88207,N1(C(C2C(C)(C)C2)=O)CCC2CC1CN2C(=O)CNC(=O)CC1CCCCC1 88208,C(=O)(CC1=CCCC1)NCC1(O)CC(NC(C=Cc2ccc(SC)s2)=O)C1 88209,C1(C(N2C(C(C)NC(c3[nH]cc(C(C)=O)c3)=O)CCCC2)=O)C(C)(C)OC1(C)C 88210,Cc1cc(C(N2CCN(C(=O)CCc3ccc(Cl)s3)C3CC23)=O)c(N)cc1F 88211,C(C(=O)NCC1CCCN1C(=O)CC1OCCO1)(C(C)C)n1cc(C)nc1 88212,C#CCC(CC(=O)NCCN(C(C)C)C1CC1)NC(C1C2CCCC12)=O 88213,C(=O)(C(C)(CNC(=O)OC(C)(C)C)OC)NCCC1CN(C(COC)=O)C1 88214,CC(c1cccnc1)=CC(=O)NC1CCN(C(c2conc2C)=O)CC1F 88215,Cc1cc(C(N2CCC(C(N3CC(C(=O)OC(C)C)C3)=O)C2C)=O)c(C)nn1 88216,N1(c2nccc(N(C)C)n2)CCC(O)C(C(N2CCCC(CS(C)(=O)=O)C2)=O)C1 88217,C(CCN=C(NCC(C(C)C)c1ccnn1C)N1CCC(C(C)(C)C)CC1)SC 88218,CC1CC(CC(=O)OC(C)(C)C)CN1C(=O)OC1(C)CN(C(=O)CSC(C)(C)C)C1 88219,C(=O)(C(C)P(C)(C)=O)NC(CNC(C(C)(F)F)=O)C(C)(C)C 88220,N1(C(C(CC)O)=O)C(C(=O)NCCc2ccc(C)s2)CC2CCCCC12 88221,C(CO)(C(=O)N1CC(CN(C)CCF)C1)O.C(=O)(CCNC(=O)CO)OC 88222,CN(C)NC(=O)CCC(=O)NCCOC1CN(C(C23CCCC2CC3)=O)C1 88223,c1(OC)c(C(=O)NCC2CCC(F)(CNC(c3cccc(Cl)c3)=O)C2)cnn1C 88224,C1(C(N(C2CCN(C(=O)C(=O)N3CCCC3)C2)C)=O)CCc2cncn2C1 88225,C1(CCNC(c2sc(F)cc2Cl)=O)CCCN(C(c2ccc(CCO)cc2)=O)C1 88226,C(=O)(CC(C)(F)F)NC(C=CC(=O)N(CCCC#C)CC)(C)C 88227,c1(CC(N2CCC3CN(C(c4c(C)coc4)=O)CC32)=O)coc2cc(O)ccc12 88228,Cc1cncc2cc(C(=O)NC3CCCCC3N(C)C(c3cc(Cl)cs3)=O)sc12 88229,Cc1ccnc(O)c1C(=O)N(CC(O)CN(C(=O)CC1(N2CCCC2)CC1)C)C 88230,N1(C(c2ccc(Cl)cc2)=O)CC2C3CCC(C2C1)N(C(C1CC1C(F)(F)F)=O)C3 88231,Cc1c(N)ccc(C(=O)N(C)CCN(C)C(C2(C)CCCC2C)=O)c1C 88232,N1(C(CNC(CC)=O)=O)CCCC2C1CCCCN2C(=O)C(O)C(C)C 88233,CC(O)CCCCCC(=O)N1CC2(C1)CN(C(c1cc(C(F)F)cc(F)c1)=O)C2 88234,C=CCCCCCCC(=O)NC1CCC(NC(=O)C=C(C)c2ccccc2F)C1 88235,N1(C(CCc2ccc(COCCC)cc2)=O)CCn2nc(CC)nc2C1 88236,c1(C(=O)NCCCC(=C)C)ccc(CNC(C2(C)CCOC2C)=O)nc1 88237,c1(C(=O)NC2CN(C(COC(CC)(C)C)=O)CC2(C)C)nccc2cccnc12 88238,C1(CNC(=O)CCc2nccs2)CN(C(C2CC2F)=O)CCC12CCOC2 88239,c1(CC(N2CCC3CN(C(C4CC4C4CC4)=O)CC23)=O)cc(Cl)cc(Cl)c1O 88240,N1(C(c2ccc(C(F)F)o2)=O)CCC2CCN(C(=O)CCc3cccs3)C2C1 88241,CC1CN(C(c2cc(O)nc(O)n2)=O)CCCN1C(=O)C(c1ccccc1)F 88242,c1(OCC)cc(F)c(NCC2CCN(c3cc(N4CCCC4)ncn3)C2)c(F)c1 88243,C1(C(=O)NC2C(NC(c3cn(CCC4CC4)nn3)=O)CCC2)CC12CCOC2 88244,CCCC(C(C(=O)NC1CCC1)N1CCCC(C(O)C(F)(F)F)C1)OC 88245,CC1CN(C(=O)C(=O)NCc2cnn(C3CC3)c2)CCS(=O)(=O)C1 88246,C12(C(=O)NC3(CO)CN(C(c4ccccc4Br)=O)C3)COC(CCO1)C2 88247,c1(OC)cc(F)c(CN2CCC(O)C(C(=O)Nc3ccc(C)nc3C)C2)c(F)c1 88248,C1(NC(CCC(C)=O)=O)CC2(C1)CC(C(=O)Nc1cccc(C(=O)N(C)C)c1)C2 88249,c1(C(N2C(C(C)C)CN(C(=O)C(=O)C(C)(C)C)CC2)=O)cn2cccc(Cl)c2n1 88250,c1(NCCOCCNC(c2ccco2)=O)cccc(Cl)c1.O=C1CCN1 88251,c1(C(=O)NC2CC(NC(C3CC3Cl)=O)C2)ccccc1.CC 88252,c1(C(=O)OC(c2c(OC)cccc2)C)c(C)ncnc1O 88253,N1(C(c2nn(C)c(C3CC3)c2)=O)CCC(NC(C2CC3CCC3C2)=O)C(CO)C1 88254,c1(C(=O)NC2(C)CC(NC(c3c(OCC)cccn3)=O)C2)ccc(C#N)cn1 88255,N1(C(C(=O)NC2(CNC(CC#N)=O)CCOC2)N2CCCC2)CCS(=O)(=O)CC1 88256,N1(C2CCN(Cc3cc(OC)cc(O)c3)C3(C2)CC3)CCc2c(Cl)cccc2C1 88257,N1(C(CCC(N)=O)=O)CCC(C2CCCN(C(C3CC4(CCOCC4)C3)=O)C2)C1 88258,N1(C(C2CC(=C)C2)=O)CCN(C(CC(C(C)(C)C)OC)=O)CC1CCCC 88259,CN1CCCC(NC(=O)NNC(=O)C2CCC(=O)N2)CC1 88260,Cc1c(Cl)c(C(N2CC3CC2CN3C(=O)Cc2cncnc2O)=O)nn1C 88261,CCC(N=c1[nH]c(=NC(C)c2ccncn2)c2ncccc2[nH]1)c1ccncc1 88262,N1(C(C(OC)OC)=O)CCC(N(C(c2ccc(C(F)(F)F)o2)=O)CC2CC2)CC1 88263,c1(C(N2C(CNC(C3CCC3)=O)CC2)=O)csnc1C1CC1 88264,C1(C2(O)CCOC2)(C(=O)Nc2cc(OC)c(NC(C)C)cc2)CC1.C(=O)C(C)(C)C 88265,c1(OCC(N2CC(NC(c3c(C)csc3)=O)C(C)(C)C2)=O)ccc2c(c1)CCC2 88266,C1(NC(CCN(CCC)C)=O)CCC2CCN(C(=O)CC3CNC(=O)C3)C12 88267,C(=O)(CC(O)CC(C)(C)C)N1CCC(=C)CC1C(=O)NOCC1CCC(OC)CC1 88268,C1(N(C(c2c(C)nc(CNC(C3(C)CC(=C)C3)=O)o2)=O)C)CCOC(C)(C)C1 88269,C(C)(CCC(C)(C)C)(C(=O)O)NCc1ccc(C(C)(C)C)o1 88270,C=C(COC(=O)C(=O)N(CC(F)(F)F)C(C)=O)CCC1CCCCC1 88271,Cc1ccccc1-n1ccc(C(=O)NC2(CN(C)C(c3[nH]cnc3C)=O)CC2)n1 88272,Cc1nnccc1NCCNC(N1CCOC(C2CC(F)(F)C2)C1)=O 88273,Cc1nc(C)n(CC(N2CC(CCNC(C3(CC(C)C)COC3)=O)C(C)C2)=O)n1 88274,c1(C(=O)NCC2C(CNC(C=CCCC)=O)C2)c(Cl)cncc1Br 88275,c1(OC)ncc(NC(C2CCN(C(=O)CC3CC(OC)C3)C2C)=O)cn1 88276,N1(C(C2C(NC(COCCOC)=O)CC2)=O)CCCC(NCCO)C1 88277,C1(NC(Cc2coc(C)c2C(F)(F)F)=O)CCN(C(=O)CN(C)C(N)=O)C1(C)C 88278,c1(C(N(C(C)CNC(=O)C(O)C2CCC2)CC)=O)cccc(-c2nc(=O)o[nH]2)c1 88279,c1(C(N2CCC(NC(CSCC=C)=O)C2(C)C)=O)ccc(C)c(C)c1O 88280,CC(CNC(=O)CC1CCOC1(C)C)CC(=O)NCCC1(C)CCCC1 88281,C1(NC(C2N(C(C(C)NC(=O)OC)=O)C3(CC2)CC3)=O)CCN(C)CC1C#N 88282,O=C1CC2C(C(N3CCCC(CCNC(c4ccc(Cl)s4)=O)C3)=O)C2C1 88283,CN1CC(NC(C2CCC2NC(=O)CCN2CCOC2=O)=O)CC1=O 88284,N1(C(=O)Nc2cc(C)c(Br)c(C)n2)CC2CC3CCCN3C2C1 88285,c1(COC)cc(C(N2CC(NC(=O)CC3(CN)CC3)C(C(N)=O)C2)=O)c(C)o1 88286,CC(C)C#CC(=O)NC(C)C=CC(=O)NCC1(C)COCCO1 88287,[N-]=[N+]=NCCCCCCNC(=O)C(C1(O)CCCCC1)NC(=O)CCC1CC1 88288,CCCC(C)(O)CC(=O)NCCCN(C)C(c1cc(Br)cnc1N(C)C)=O 88289,c1(OC)cc(C(N2CC(OC)CC2CNC(c2ccc[n+]([O-])c2)=O)=O)cc(Cl)n1 88290,c1(OCC)cccc(CCC(c2nnnn2C)NCCCS(=O)(=O)N(C)C)c1 88291,N1(C(=O)C#CC2CC2)C2CCC1CN(c1c(Cl)cncc1[N+](=O)[O-])CC2 88292,n1(CC)ncc(C(N2CC=CC(NC(=O)C(C)NC(C3C=CCC3)=O)C2)=O)c1C 88293,c1(C(=O)NC2CC(O)(CNC(CCNC(=O)C3CC3)=O)C2)cnc2c(c1)COC2 88294,N1(C(CN(C(C)C)C)=O)CCC(CCCNC(=O)CCc2ccc(F)cc2)CC1 88295,C1(C(=O)NCCCOCCN(C(c2cn(CCC)nn2)=O)C)CCCOC1C 88296,C1(CNC(c2nc(CNC(CNC(C(C)(C)C)=O)=O)oc2)=O)CC[Si](C)(C)C1 88297,C12(C(=O)NCCCCC(C)NC(C(C)c3ncco3)=O)CC3CC(CC(C3)C1)C2 88298,c1(C(=O)OC)ccc2oc(CNc3nccc(C)n3)cc2c1 88299,N1(C(CCC#CC)=O)CCC2(CC1)OCCC2NC(c1cc(OC)cs1)=O 88300,c1(C(N2CC3C(CCNC(c4c(C)cco4)=O)(CC3)C2)=O)cccc([N+](=O)[O-])c1 88301,C1(NC(C2CN(C)C2)=O)CN(C(C2(O)CCCC2)=O)CCC1F 88302,N1(C(c2ncc(C)cc2F)=O)CC2CC(NC(=O)C(C)C)CC2C1 88303,CC1(C)CCCC(CNCCCn2ncc3ccccc23)CC1 88304,c1(OC)cc(C(=O)NCC(CNC(=O)C(O)C(C)C)C(F)(F)F)cc(N)c1O 88305,C(=O)(C(F)(F)C(F)F)N1CCC(C(C)NC(=O)CC2CSC2)C1 88306,C12(C(=O)NCC3CC(NC(=O)Cc4cccc(O)c4)C3)CSCC1C2(F)F 88307,c1(OC)ccc(C(=O)CCC(=O)N2CCCC2(C)CNC(c2nncs2)=O)cc1 88308,C1(CCCC)CCC(C(=O)NCCC2CN(C(=O)CCOC)CCO2)CC1 88309,C1(C(C(N2CC(C)C(NC(c3cscc3C#N)=O)C2)=O)O)CCS(=O)(=O)CC1 88310,Cc1cnn2cc(C(N3CCCC3CN(C(=O)CCSCC(N)=O)C)=O)cnc12 88311,c1(CC(N2CC(NC(Cc3c(C)cco3)=O)(CO)C2)=O)cccc2c1OCCO2 88312,c1(CC)cc([N+](=O)[O-])ccc1N(CCNC(=O)C(C)C(C)(C)C)C1CC1 88313,C12(NC(C(C)(F)F)=O)CC1CN(C(c1csc(Cl)n1)=O)C2 88314,C1(CC(N2CC(OC)(CNC(=O)CC(=O)NC3CC3)C2)=O)CCN(C)CC1 88315,c1(CC)[nH]c(=N)sc1C(=O)N(CC(C)N(C)C(c1cncnc1C)=O)C 88316,N1(Cc2c(C)nc[nH]2)CCc2nc(C(=O)NC3CCC(N(C)C)CC3)cn2CC1 88317,N1(C(C=Cc2n(CC)ccn2)=O)CCCC2(NC(=O)C=CC(=O)OCC)CC2C1 88318,c1(C(C(=O)NC)N(C)Cc2ccco2)cccc(OC(F)(F)C(F)Cl)c1 88319,c1(C(N(CC(O)CNC(=O)C#CC2CC2)C)=O)cnc2c(F)c(F)ccc2c1 88320,c1(C(N(CCC(C(C)C)NC(C(C)OC)=O)C)=O)cccc2ncc(Br)n12 88321,C1(C(=O)NC(C(=O)OC)CC2CC2)CCCN(C(c2cc(OC)n(C)n2)=O)C1 88322,CCC(C)(C)CC(=O)N1CCC(C(N2CC3C(C(N)=O)C3C2)=O)CC1 88323,c1(NC(C)=O)cccc(C(=O)NC2CCCC(CNC(c3scnc3Cl)=O)C2)c1 88324,c1(C(=O)NC(C2(O)CCN(C(c3ccn(C)c3)=O)C2)C)cc2c(ccn2C)[nH]1 88325,N1(CC(=O)NC(C)(CNC(=O)Cc2csc(C3CC3)n2)C2CC2)CCOCC1=O 88326,N1(C(C(CN(C(CN(CCC#C)C)=O)C)(C)C)=O)CC2OCCN(C)C2C1 88327,N1(C(CSc2c(C)cccc2)=O)CCC2(CCN(C(C3(C)CC4CC4C3)=O)C2)C1 88328,c1(C(=O)NC2CCC(NC(c3c(OC)cc(Cl)nc3)=O)C2)cc(C)c(F)cc1Br 88329,c1(C(C(=O)NCC2(C)N(C(c3onc(CC)n3)=O)CCC2)C)cc(C)cc(F)c1 88330,C1(C(=O)NC(C)(C)CNC(C2CC(C)(F)C2)=O)CCCC1(F)F 88331,c1(C(N2C(CCNC(=O)C3=CCCCC3)CCC2)=O)cc2cccn2cn1 88332,C#CC1CN(C(c2cnn(C(C)C)c2)=O)CCN1C(=O)C(c1ccncc1C)C 88333,CCC(CC(C)C)C(=O)N1CCC(C(C)CNC(=O)C(C)(C)c2nccs2)CC1 88334,c1(CNC(C=CC)=O)nn(C)c2c1CN(C(c1ccnc(C)c1)=O)CC2 88335,C1(C(=O)NCC(CCNC(=O)CCc2cnco2)O)CCc2ccccc2C1 88336,C1(C(=O)NCC2(O)CC(NC(Cc3ccc(C)o3)=O)C2)CCCCN1S(N)(=O)=O 88337,C1(CN(C)C(c2csc(=N)[nH]2)=O)CCCC(NC(=O)C(=O)Nc2ncc[nH]2)C1 88338,c1(C(=O)OCC)cnc(OC)cn1.C12CC3(C1)CC3N2.c12[nH]nc(c1Cl)NC2=O 88339,C1(C(F)(F)F)(C(=O)NC(CC)CNC(c2ccnnc2)=O)CC=CCO1 88340,N1(c2nccc(OC)n2)CCC(O)(C(=O)NC2CCNC2=O)CC1 88341,N1(c2nnc(C)s2)CCOC2(CCN(C(c3ccc4ncnn4c3)=O)CC2)C1 88342,N1(C(CC=CC)=O)CCCCC1CCN(C(=O)C(C(=O)OC)OC)C 88343,c1(CC)nn(C)cc1CNC(C1COCCN1C(=O)C=C=C(C)C)=O 88344,N1(C(CN(CCC)C)=O)CCC(NC(c2ccc(OC)nc2C)=O)C12CCCC2 88345,N1(C(C=CCC)=O)CCCCC1CN(C(C1(C)COC1)=O)CC 88346,N1(C(c2cc(CCNC(c3cnc(C)o3)=O)on2)=O)CCOC2CC12 88347,c1(CC(CNC(C2CCCCC2)=O)NC(=O)CCC2CCCO2)ccccc1 88348,C1(CC)CC(C(=O)NCC(C)CC(=O)OC)CCN1C(c1c[nH]c(=N)c(C)c1)=O 88349,N1(C(CSCC#C)=O)CCC(O)(CCNC(=O)C(c2nc(C)cs2)C)C1 88350,C1(C(=O)NCCC2CN(C(C3CC(C4CC4)C3)=O)C2)(CC)CCCCO1 88351,C1(C(N(CC)CC2CCCO2)=O)C2CN(C(=O)CC3COCCO3)CC12 88352,N1(C(CC2CCN(C(C3C(CCC)CCC3)=O)C2)=O)CC(OCC)C2(CC2)C1 88353,n1(CC)nc(C(=O)NCC2CC(NC(=O)C(C)(COC)OC)C2)c(C)n1 88354,n1(CC)cnc(C(=O)NCC2(NC(c3ccn(CC(C)C)n3)=O)CCCC2)n1 88355,c1(C(=O)NCCn2ccnc2)cc2ccc(-c3cnn(C4CC4)c3)cc2s1 88356,N1(C(c2c(C)noc2N)=O)CCC2(CCC(NC(=O)Cc3cocn3)C2)CC1 88357,C1(C2CN(C(=O)C(F)C(F)(F)F)C2)(NC(c2cccc(-n3cccn3)c2)=O)CC1 88358,c1(C(N2CC(C)C(O)C2)C(=O)NC)cccc2c1CCO2.c1(C2CC2)ccccc1.CC 88359,N1(CC(=O)NC2CC(CC(=O)N(CC(C)(C)CO)C)C2)CC(=O)NC1=O 88360,c1(CC(N2CC(NC(C3N(CC)CC3)=O)C(O)C2)=O)cc(C)ccc1OC 88361,C1(C(N2C(CC)CN(C(=O)CCCF)CC2)=O)CCC(C2CC2)CC1 88362,C1(C2CCN(C(=O)Cn3nccn3)C2)CCCCN1C(c1cccc(OC)n1)=O 88363,C#CC1(O)CC(C(=O)NC2(C(=O)NCCNS(=O)(=O)CC)CCSC2)C1 88364,CCC(C(=O)NCC1(OC)CC1)N(C(=O)C(C)(F)c1ccon1)C 88365,c1(NC2(C)CCN(C(C(C=CC)O)=O)C2)ncc(C(=O)OCC)cc1[N+](=O)[O-] 88366,C1(NC(=O)C2CC2)CCCC1C(=O)NC1CC(F)(F)C1 88367,CC(CNC(C1CN(C)CCN1C)=O)C(F)C(=O)NC1CCNC(=O)C1 88368,c1(NCC(CC)(C)OC)ccc(S(=O)(=O)NCC(C)(C)CC2CC2)c(Cl)c1 88369,c1(C(=O)NC2CCC(CNC(CS(N)(=O)=O)=O)C2)cnc2nccn2c1 88370,C1(CNC(CSCC(C)C)=O)COC(CNC(=O)COCCC(C)C)C1 88371,C1(C(=O)NC(C2(CNC(c3cc(C)n(C)c3)=O)CC2)C)CCC(C)(C)OC1 88372,N1(C(COCCOC)=O)CC2CC2(C(=O)NC(CO)C(=O)O)C1 88373,N12CC3CC1CN3C(=O)C(O)C1CN(C3CN2C3)C1.C(=O)NC 88374,N1(C(C2(C#C)CCCC2)=O)CCC2(CCCC2CNC(C2CCNC2=O)=O)CC1 88375,N1(C(=O)OCC)CSCC1CCN(C(=O)CC1CCC(=O)O1)CC.c12cn-1nn2 88376,C1(NC(C(CNC(C(C2CCC2)OC)=O)OC)=O)CC(C)(C)C12CCC2 88377,N1(C(C(=Cc2cnc[nH]2)C)=O)CC2(CCN(C(=O)CC(C)(C)C(=O)OC)C2)C1 88378,CC1OC2(C(=O)NC3CCN(C(c4cc(C(N)=O)co4)=O)C3)CC1C2 88379,C#CCCCCC(=O)NC1CCC(NC(C2(CCOC)CC2)=O)C1 88380,CCC(CC)CCC(=O)NCCCN(C(c1cc(OC)ccc1CC)=O)C1CC1 88381,Cc1ccn2cc(CN3CCCCC3CNC(=O)OC(C)(C)C)nc2c1 88382,N1(C(C2N(CC)CC2)=O)CCC(CNC(=O)C=CCN(CC)CC)C1(C)C 88383,N1(C(C=CCOC)=O)C2CCCC1CC(NC(C1CC(n3cnnc3)C1)=O)C2 88384,c1(C(c2nnc(N3CCC(C)C3C)n2CC(C)C)[N+](=O)[O-])cc2ccccc2o1 88385,C1(F)(C(N(CCCNC(C2(F)CCOC2)=O)C)=O)CCCCC1 88386,CC1(C)CCC(NC(C2(C)CC2)=O)C(CNC(=O)C(F)(F)C2CCC2)C1 88387,c1(C(=O)NC2C(CNC(c3cnc4c(c3)CCC4)=O)C2)cccc2c1COCC2 88388,C1(C(N2CCC(N(C(C(C)=CC)=O)C)C2)=O)CC2CCC(C1)C2F 88389,N1(CC(=O)NCC2C(C)CN(C(=O)C=CC3CCOC3)C2)CCCCCCC1=O 88390,Cc1cc(F)ccc1C(=O)N(C1C2CN(C(C3CCCOC3C)=O)CC12)C 88391,CCC(C)(C(=O)N(C)CC1CCN(C(c2ccccc2OC)=O)CC1)C(F)F 88392,CN1CCC2CCC(C1)N2C(=O)CCC1CCC(NC(=O)C2=COCC2)C1 88393,C1(CNC(C2(C)ON=C(C)C2)=O)CN(C(=O)CC2(C)CC(F)(F)C2)CC12CCC2 88394,N1(C(C(=O)NC(CC)C)CCC2CC2C)CC(C(=O)OC)C(C2CCCCC2)C1 88395,c1(NC(C(F)=CC)=O)ccc(NC(c2cc(CC(C)C)c[nH]2)=O)cc1C 88396,N1(C(C(C)C(C)(F)F)=O)CCC(C2(O)CN(C(=O)CNS(N)(=O)=O)C2)CC1 88397,N1(C(C(=O)NCC)=O)CC2CC1(CNC(c1ncc(C(F)F)s1)=O)C2 88398,c1(CC(=O)NCCN(C(C(C=CCCC)O)=O)C2CC2)ccc(C)cc1Cl 88399,c1(OC)ccc(F)cc1CC(=O)N(C1CCCN(C(C2CCCO2)=O)CC1)C 88400,C(=O)(C1CCOc2ccccc21)N1CCC(NC(C(C)NC(N)=O)=O)CC1 88401,CC(F)(F)CCCC(C(=O)NCCC1CC1)N1CCC(OC2CCC2)C1 88402,c1(C(N2CCC(N3CCOC3=O)C2)C(=O)NCCOC)cnc(OC)c(Cl)c1 88403,C(=O)(C#CC1CCCC1)NC(CCC)C(=O)NC1CC(CC(C)(C)C)C1 88404,c1(C(=O)NC(CCN(C(c2cc(=NC)[nH]cc2)=O)C)C)cnc2c(c1)COC2 88405,N1(C(C(CCC)F)=O)CC(CNC(c2c(C)noc2C2CC2)=O)CC(C)C1 88406,C(CO)(C(O)c1cccnc1)NC(c1nc(Br)c[nH]1)=O 88407,c1(OCC(N2C3(CNC(C4N(C)C(=O)OC4)=O)CC(C2)C3)=O)ccc(Cl)cc1F 88408,C(C(C(C)(C)C)NC(=O)C=CCOC1CCOCC1)NC(COCC=C)=O 88409,CCC(C)C(=O)NC(C)CCCNC(c1cnoc1-c1cccs1)=O 88410,CCCCCC(C)C(=O)N1CCN(C(=O)COc2ccc(Br)cc2)CC1C#N 88411,C(=O)(C(F)C(F)(F)C(F)(F)F)NC1C(CNC(C(=O)N(C)C)=O)CC1 88412,N1(C2CN(C(C=CC(C)C)=O)C2)CC(NC(=O)C(=O)N(C)C)CC1=O 88413,C1(NC(=O)CCc2cc(C3CCC3)on2)(CO)CCN(C(=O)CC(F)F)C1 88414,c1(C(=O)NCC=CCNC(C2C(SCC)N(C)CC2)=O)n[nH]c2c1CCCCC2 88415,C1(CNC(C(=O)NCC2CC(C)(C)C2)=O)Cc2ccc(Br)cc2C1 88416,C1(C(=O)NCCN(C(C2CCCN2C(=O)OC)=O)CC)(C)CC(F)(F)C1.CC 88417,c1(NC)cnncc1C(=O)NCC1CCC(NC(c2cc(O)ncn2)=O)C1 88418,CC(CCC(C)(C)C)C(=O)NCC1CC2COCC2N1C(=O)CCN(C)CCO 88419,C1(CC(N2C3C(NC(c4cc[nH]n4)=O)C(C3)C2)=O)Cc2ccc(Br)cc2C1 88420,CCC(CC)CCCC(=O)N1CCCC1C(N1CCCC(N=[N+]=[N-])C1)=O 88421,C1(NC(c2cc(C(N)=O)[nH]c2)=O)CC2CCC1(NC(C1CC=CC(O)C1)=O)C2 88422,C(=O)(C1c2c[nH]nc2CN1C(=O)C#CC1(C)COC1)N(CC(C)O)CC1CC1 88423,c1(CC)c[nH]c2ncnc(N3CCC(CF)(NC(C4C=CCC4)=O)C3)c12 88424,O=C1CCCC(C(N2CCCC(NC(c3cnn(C4CC4)c3)=O)C2)=O)CC1 88425,CON(C)C(=O)C(C)NC1CCCCC1n1cc(CC(C)(C)C(=O)O)nn1 88426,N1(C(C(C)C2CC2)=O)CC2(CCC(CNC(=O)Cc3ccc(Cl)c(F)c3)O2)C1 88427,c1(C(N2C(CNC(CNC(C)=O)=O)C(C)CC2)=O)ccc2n[nH]c(C)c2c1Cl 88428,N1(C(C2(F)C(C)C2)=O)CCOC2(C1)CN(C(=O)CCc1ccccc1Cl)C2 88429,CC1=NOC(CC(=O)NC(C)(C)CN(C(=O)C=Cc2ccco2)C)C1 88430,N1(C(c2c(CC)[nH]cc2)=O)CCOCC2(COCCN2C(=O)C(O)C(C)CC)C1 88431,CC(C)C(C)CC(=O)NC(CC1CC1)C(=O)N(C1(c2cc[nH]n2)CC1)C 88432,c1(C(N(CCC(=O)NC2CCSC2)CC=C)=O)ccnn1C 88433,c1(C(=O)NC(CCN(C(C(C)=C2CC2)=O)C)C)ccc(C2CNC(=O)C2)cc1 88434,N1(C(CC(=O)NCC)=O)CC(NC(=O)CN2CCC(C)CC2)CC1(C)CC 88435,CN1CCC(NC(N2CCCC(C)(N3CCCC3)C2)=O)C(C#N)C1 88436,c1(N(C2CCN(C(c3ccccc3Cl)=O)C2)C)cnc(C#N)cn1 88437,C12(CNC(C(CCO)N(C)C)=O)CCC1CN(C(=O)Cc1c[nH]nc1O)C2 88438,N1(C(Cc2cc(C)cc(C)c2)=O)CCC(NC(C2CC2C)=O)CC(C)(C)C1 88439,CC(C(C)(C)C)=CC(N1CCC(NC(=O)CCCc2csc(C)n2)C1)=O 88440,CCC(CO)C(=O)NC(C1(O)CN(C(=O)C(O)Cc2ccccc2)C1)C 88441,N1(Cc2c(OC)cc(Br)cn2)CCC(F)(F)C(NC(=O)Cc2ccsc2)C1 88442,C(CCC(=O)NC1CCOC2(CCC2)C1)(C(C)C)NC(C(c1ccn(C)n1)C)=O 88443,c1(CC(=O)NCC2CCCC(NC(c3csnn3)=O)C2)nc([N+](=O)[O-])n[nH]1 88444,N1(C(C2(C)CCOC2)=O)CCN(C(=O)CCCN=[N+]=[N-])C(CC(F)(F)F)C1 88445,c1(N(CC(C)C)C)ccc(C(N2CC(F)(CNC(C3CC3C#N)=O)C2)=O)cc1 88446,C1(N(C(=O)CCN2CCOCC2)C)CCC2CN(C(c3ccoc3Cl)=O)CC12 88447,n1(CCCN(C)C(C2(C3CCCCO3)CC2)=O)cc(C2CCCO2)nn1 88448,O=C(CC1=CCCCC1)N1CCC(O)(CNC(=O)C(CCl)c2ccccc2)C1 88449,C1(CNC(C(CC=C)NC(=O)C2=C(Cl)CC2)=O)CCCC12CCC2 88450,C1(OC)(CNC(=O)C=CC(F)(F)F)CCN(C(=O)C(C)(C)CF)CC1 88451,CC(O)(CNC(c1conc1CNC(C1(CO)CCOC1)=O)=O)C(F)(F)F 88452,c1(C(N2CCC(N(CCC)C(c3ccc(C)cc3)=O)C2)=O)cc(F)c(N)cc1F 88453,c1(C(=O)NC(C(C)NC(CS(CC)(=O)=O)=O)(C)C)cccc2cc(O)ncc12 88454,C1(C(=O)NCCCc2cn(CCC(F)(F)CO)nn2)CCC(C(F)F)CC1 88455,C1(C(=O)NCc2scc(C)c2)C2CC1N(C(=O)CCc1ncccn1)C2 88456,c1(CC(=O)NC2CC3CC(NC(C(C)OCC=C)=O)C3C2)c(C)cc(C)nc1O 88457,CN1CCN(C2CCCC2c2ccc(CNC(c3ccccn3)=O)cc2)CC1 88458,c1(C(=O)NC2CCN(C(CC)=O)CC(C)(C)C2)ccc2c(c1)COCCN2 88459,N1(C(CCOCC#C)=O)CCC2CN(C(C3OCCN(C)C3=O)=O)CC12 88460,C1(CC)CCCN(C(C2CC(C#N)(OC)C2)=O)C1C(=O)NC1CCN(OC)CC1 88461,c1(N2C(=O)CC(C(=O)NCC(CN(C(=O)C(C)(C)O)C)O)C2)ccc(F)c(F)c1 88462,C1(C(=O)NC(C2CC2NC2CC(CC3CC3)C2)=O)COCCN1CC1CCC1 88463,C1(C(=O)NCCOCC2CC2)(CNC(C(C)OC2CCCC2)=O)CCCO1 88464,C(=O)(CS(=O)(=O)C1CC1)NC1C(C2CCN(C(C(F)=C(C)C)=O)CC2)OCCC1 88465,CN1C2CCC1CN(C(C1COCCN(C(C3CCCO3)=O)C1)=O)CC2 88466,c1(N(C(c2cnc(C)[nH]2)=O)CC2CC2)ccc(Cl)cc1 88467,C(CCC(C)(C)NC(c1cnc[nH]1)=O)NC(c1cn(CC(CC)O)nn1)=O 88468,CC1(C(=O)Nc2cncc(Br)c2Cl)CCCN(C(=O)CCc2cnccn2)C1 88469,c1(C(=O)NC2CCN(C(CSCCCC)=O)CC2)ccnc2c1ccn2C 88470,N1(C(Cc2c(C)nccc2)=O)CCC2CCC12CNC(c1c(C)[nH]c(C)c1C)=O 88471,C(=O)(CS(=O)(=O)CCO)NCC1(CO)CCN(C(C(COC)O)=O)C1 88472,C(CCCC(C)NC(c1cnn(CC)n1)=O)NC(C(C)(C)OCC)=O 88473,c1(NC(C)CCc2ccccc2F)nccc(=NCC2(CCO)CC2)[nH]1 88474,c1(C(C)OC(CC(C)C)C)nc(-c2cnn(C)c2)nn1CC1CCC1 88475,N1(CC(=O)NCC(N(C(CCCCC#C)=O)C)C2CC2)CCc2ccccc21 88476,C1(C(=O)NCCc2ccc(F)cc2)CCN(Cc2ccc(F)cc2O)CC1O 88477,N(C(=NC1CCS(=O)(=O)C1)NCC1CC(C)(C)C1)C1C(OCC)C1 88478,C#CCCCCCC(=O)NCC1C2CN(C(=O)CC(C)N(C)C)CC12 88479,S(=O)(=O)(CC(=O)NC1CCCC1NC(c1nccn1C(C)C)=O)NC 88480,C1(CC(=O)N(CCCC=C)C)CCCN(C(C2CCCN2CC)=O)CC1 88481,C(=O)(C1CCCc2ncnn21)N1CC(O)CC(NC(C2(C)CCCCC2)=O)C1 88482,Cc1nn(CC(=O)NC2C3CN(C(=O)C(C)CC4CC4)CC23)c(C)c1Cl 88483,Cc1cc(C(=O)N(C)CCc2cn(C(C)C(C)O)nn2)n2nccc2n1 88484,c1(CC(N2C(C(=O)OC)C=CCC2)=O)ccc(S(=O)(=O)NC(=O)C2CC2)s1 88485,N1(CC(=O)N(S(CC)(=O)=O)CC)CCCC(NC(=O)CC(F)F)C1 88486,Cc1n[nH]c2cnc(C(=O)NCC(C(C)C(C)C)NC(c3nocc3Cl)=O)cc12 88487,N1(C(COC(CC)C)=O)CC(NC(c2cn[nH]c2)=O)C(C2CC2)C1 88488,C1(CC)CC(C(=O)NCc2cccc(Cl)c2)CCN1C(c1ccn(C2CC2)n1)=O 88489,N(C1CCCc2cc(CNC(=O)C=Cc3ncco3)ccc21)C(CCOC)=O 88490,C1(OC)(OC)CCC1C(=O)NC(C)C(=O)NCC1C(C)C1C 88491,C(=O)(C(=O)CCC(C)(C)C)NCC1C(C)CN(C(c2cc([N+](=O)[O-])n[nH]2)=O)CC1 88492,N1(C(COCC(=C)C)=O)CCN(C(C2CCC(=O)N2CCC)=O)CC1C(F)F 88493,N1(C(CC(C)F)=O)CCC2(CC1)CN(C(C1Cc3ccc(F)cc3C1)=O)C2 88494,c1(C(N2C(C(N(CCCO)C(C)C)=O)CC2C)=O)ccc(CO)cn1 88495,C1(C(=O)NC2(CCOC)CC2)COCCC1NC(=O)CC1CSC1 88496,Nc1ccc(C(N2CCC(O)(CNC(C3CCS(=O)(=O)N3)=O)C2)=O)c(O)c1 88497,C1(NC(CN2CCC(C)CC2)=O)CC(F)CN(C(c2cc(C(N)=O)no2)=O)C1 88498,CC(CC(F)(F)F)C(=O)Nc1ncc(C(F)(F)F)s1 88499,c1(OC)ccccc1C(C)(C)NC(=O)NCc1ncccc1C(F)F 88500,c1(NC(=O)NC2C(C)C2(F)F)cc(-n2ccnc2)ncn1 88501,C1(OCC(=O)NC(C)CCNC(=O)CC2(CO)CCOCC2)CCC(F)(F)CC1 88502,c1(-c2nc(CC(CCC)C)n(CC(C)C3CC3)n2)ccc2ccccc2n1 88503,N1(C(C(F)=CCC)=O)CCCN(C(c2n[nH]c(CC)n2)=O)CC1 88504,CC1=C(C(=O)N2CCC(NC(C34CCCC3C4)=O)CC2C)C(=O)OC1(C)C 88505,c1(CC(=O)NCCN(CCC)C(c2csc(Br)c2)=O)cc(OC)no1 88506,C1(OCC)CN(C(C2(CC)CCOC2)=O)CC1CNC(c1ncccc1NC)=O 88507,CCC(CC(F)F)C(=O)N1CCN(C(c2cscc2SC)=O)CC1 88508,N1(C(C(C=C)C)=O)C2CCC(C(N3CC4(C)CCC4(C)C3)=O)C1CC2 88509,CC(CN(C)C)N=c1[nH]c2c(c(=NC(C)c3ncc(C(F)(F)F)[nH]3)[nH]1)CCC2 88510,n1(C(C(=O)NCCN(CC(=O)OCC)CCNC(N)=O)C)cc(Br)cn1 88511,c1(CNC(CC2(OC)CN(C(C3OCCCC3(C)C)=O)C2)=O)ccnc(F)c1F 88512,c1(C(C)C)[nH]nc(C(N2CC(NC(C3(C)C=CCC3)=O)C2)=O)c1[N+](=O)[O-] 88513,N#CC1(C(=O)NCC2(NC(=O)Cc3ccccc3)CCC2)CCOCC1 88514,Cc1cc(CNC(c2conc2C(C2CC2)NC(C)C)=O)n(C)n1 88515,Cc1cnc2c(C(=O)N(C3CCN(C(=O)CC4CC(F)C4)C3)C)cnn2c1 88516,Cc1c(F)cc(C(N2CCCC(NC(C34CSC(C3)C4)=O)CC2)=O)c(F)c1N 88517,Cc1nc(C(N2CCCC(n3cc(CNC(C4CC4C#N)=O)nn3)C2)=O)c(C)o1 88518,c1(CNC(c2cc(CCNC(COCC(=C)C)=O)on2)=O)ccc(O)c(F)c1 88519,c1(N(CCC)C)ccc(C(=O)NCCN(C(C2SCCS2)=O)C2CC2)cc1 88520,C(C(=O)NCCc1cn(Cc2cc(C)no2)nn1)(C(C(C)C)OC)OC 88521,Cc1nc(CO)sc1C(=O)NCC(C)NC(c1nc(=N)cc[nH]1)=O 88522,c1(C(N(CCOCCNC(C(C(C)O)C)=O)C)=O)ccc(F)c2ccoc12 88523,Cc1nc[nH]c1CC(=O)NC(C)(CNC(c1cccnn1)=O)C1CC1 88524,C1(NC(CCC=C)=O)C=CCN(C(=O)C(C)NC(C2CCCCC2)=O)C1 88525,Cc1[nH][nH]c1C(N1CC(O)(c2cn(C(C)C)nn2)C1)=O 88526,C1(O)(CNC(c2c(CNC(c3c(C)nc(CC)o3)=O)cco2)=O)CCC(C)(C)C1 88527,C=CCC(C)(C)CC(=O)NCCCCNC(c1c(C)ncnc1O)=O 88528,C1(NC(=O)CC2CNC(=O)O2)CN(C(c2ccnc3[nH]cnc23)=O)C2(CCC2)C1 88529,Cc1cnc(Cl)c(S(=O)(=O)N2CCCC2CC(=O)Nc2ccnc(Cl)c2I)c1 88530,C=C(C)C1CN(C(C2C3CC3CN2C(c2cc(C(F)F)[nH]n2)=O)=O)CCO1 88531,c1(N2CCCC(C)(CO)C2)cc(Br)ccc1S(=O)(=O)NCc1ccnc(C#N)c1 88532,Cn1cnc2cc(C(N3CCCC(NC(=O)C4=CCCOC4)C3)=O)ccc12 88533,C1(C(C)C)CN(C(=O)CN2CCNC(=O)C2)CCN1C(=O)Cc1cccnc1 88534,C1(CC=C)(NC(C2(COC)CC2)=O)CCN(C(c2cc(=O)cc[nH]2)=O)CC1 88535,c1(C(N2C(C(N3CCCC3)=O)CC2)=O)cccc(-c2nc(O)n[nH]2)c1 88536,N1(C(C2(CCOC)CC2)=O)CCN(C(c2cn(C3CC3)nc2C)=O)CC(C)(C)C1 88537,c1(OC)cc(C(N2CCC2CNC(c2cccc3ccoc23)=O)=O)cc(N)c1N 88538,C12(C(=O)NC3CCC(NC(C4C=CCC4)=O)CC3)C3CC(CC13)C2(F)F 88539,CC1CN(C(C2(F)CC=CCC2)=O)CC1NC(c1cnc(COC(C)(C)C)s1)=O 88540,N1(C(C(C)N(C(c2csc(F)c2)=O)C2CC2)=O)CC(S(C)(=N)=O)C1 88541,N1(C(C)=O)CC2CN(C(=O)CCn3cc(-c4ccc(C5CC5)cc4)nn3)C2C1 88542,Cc1cc(F)ccc1C(=O)NCC1CCCN1Cc1cc[nH]c1 88543,C(CC(F)F)(C(=O)NC1CCCC1C#N)NC(COCCSC)=O 88544,c1(C(N2CC3CC3(NC(C34CCCN3CCC4)=O)C2)=O)ccc2nccn2n1 88545,CC1COCCN(C(=O)CCN(C(=O)COC2(C)CCC2)C2CC2)C1 88546,N1(C(CCC(=C)C)=O)CCC2(CCOC2)C(CNC(c2csc(COC)c2)=O)C1 88547,N1(C(C(CCOC)NC(=O)CCCCNC(N)=O)=O)CCNC(=O)C1C 88548,c1(C(=O)NC2CC(CNC(C(C)C3CCC3)=O)C2)n[nH]c2ccc(Cl)cc12 88549,c1(C(=O)NCCC2N(C(CC(C)NC(N)=O)=O)CCC2)nn(C)nc1Br 88550,C(C(=O)N(C)CC1CCOCC1)(C(C)CC)N(C(C1CCC(=C)CC1)=O)C 88551,CC1(C)CCOC1CS(=O)(=O)NC(c1cnc(CN2CC(N)C2)o1)=O 88552,Cc1cccc2c1CCOC2C(=O)NC1COC2CN(C(=O)C3=CCOC3)CC12 88553,C(=O)(CC(C)(C)C(=O)OCC)NC1C(NC(CCC=C)=O)CC1 88554,C=Cn1ncc(C(N2CCC(C)(C)C2CC(=O)NC2(C)CC(C)C2)=O)c1N 88555,C1(CNC(CCCC(C)=O)=O)CN(C(=O)C(C)(C)C2CCCCO2)CCC1(F)F 88556,c1(OC)coc(C(=O)NC2CC(CCNC(=O)Cn3cc(C#N)cn3)C2)cc1=O 88557,C(CC(C)(C)C)(C(=O)N1CC(C)CCC1C(=O)NCC(N1CC=CC1)=O)OC 88558,C#Cc1cccc(C(N2CC(CNC(c3cnn4ccn(C)c34)=O)C2)=O)c1F 88559,c1(C(N(CC(CN(C(=O)CCC2CCCO2)C)O)C)=O)nccc2cccnc12 88560,CCCCCC(F)C(=O)N1CC(NC(=O)CCCCCn2cnnn2)C(C)(C)C1 88561,C1(N(C(C2C(C#C)C2)=O)C)CCCN(C(c2cc(C)n(-c3ccccn3)n2)=O)C1 88562,N1(C(CC)CC)CC(C(=O)NC2CCC(CNC(=O)C(F)CC)CC2)CC1=O 88563,c1(C(=O)NCC2(O)CN(C(CC3CC(=O)OC3)=O)C2)cc(C2CC2)ccn1 88564,C(=O)(CC(C)(F)F)N1C(C2(CCC(=O)NC3(C)CCC3)CC2)CCC1 88565,C1(NC(C(CC)NC(C)=O)=O)CCC2CC1CN2C(=O)C(C)OCCC(C)C 88566,N1(C(C(CC)(F)F)=O)CCc2ccccc2C(NC(c2ccncc2Cl)=O)C1 88567,C1(C)(NC(CC2C=CC(NC(c3cc(C(C)C)on3)=O)C2)=O)CC(F)(F)C1 88568,c1(C(C)=O)[nH]c2ccccc2c1C(=O)NCC1CC1F.C12CCCC1NC2=O 88569,Cc1ncnc(C(=O)NCC(CC2CC2)C(=O)NC2(c3nn[nH]n3)CC2)c1C 88570,C12(C(=O)NC(CCC)c3nn[nH]n3)CCN(C(=O)CSC(F)(F)F)CCC1C2 88571,C(=O)(C(O)CCCNC(C)=O)NCC(C1CCCCC1)OCC(C1(C)CCC1)=O 88572,C1(CC2(C)CCCN2Cc2coc([Si](C)(C)C)c2)CCc2ccc(O)cc2C1 88573,N1(C(=O)NC2CC(c3ccccc3)(OC)C2)CCCc2cc(C(N)=O)ccc21 88574,CC(C(=O)NC1CC(CC(N2CCOCC23CC3)=O)C1)S(N)(=O)=O 88575,C1(C)(c2cn(-c3ncn(C)n3)nn2)COCCN1C(c1nc(I)cs1)=O 88576,C(=O)(C1CCCc2ncnn21)N1CC(=C(CNC(c2csc(S)n2)=O)F)C1 88577,C(CC(C(C)(C)C)NC(=O)CC1CN(C(C)=O)C1)N(C(C(COC)(C)OC)=O)C 88578,N1(C(c2ccnc(F)c2Cl)=O)CC(CO)C2(CCN(C(C3CC34CC4)=O)CC2)C1 88579,c1(C(N(CCCN(C(=O)CCc2ccnc(Cl)c2)C)C)=O)cnn2ccn(C)c12 88580,C(=O)(C(C)(C)C(C)C)NCCC(N1CCC(N(C(CCCOC)=O)C)C1)=O 88581,c1(COC(CC2ON=C(CC)C2)=O)ccc2c(c1)CCCO2 88582,c1(OC)ccc2c(c1)CC(C(=O)NCC(C(C)C)NC(c1c[nH]nc1F)=O)CC2 88583,c1(NC(C)=O)ccc(C(=O)NC2CC(CNC(C3CCSCC3)=O)C2(C)C)cn1 88584,C(=O)(CCC(=O)N1CC(CC(C)NC(=O)CCCC2CC2)C1)NCCC 88585,Cc1cc(C(N2CCCC2(C(=O)N(C(CO)C2CC2)C)C(C)C)=O)nc(O)c1 88586,c1(CCN(C(=O)CNC(=O)CN(C)CC2(CO)COC2)C)ccccc1 88587,N1(C(C(C)n2ccnc2)=O)CCC(O)C(NC(c2cc(=O)cc(Cl)[nH]2)=O)C1 88588,CCCCC(CC(=O)N1CCC(CO)C12CCC2)NC(=O)CCC(C)(C)F 88589,S(=O)(=O)(c1ccc(NC2CCC(CO)C2)cc1Cl)NCCc1nc(C)sc1 88590,N1(C(C(CC)OC2CCCC2)=O)CCCC(CC(=O)N(C)CC2(F)CCC2)C1 88591,N1(C(CCCOCCC)=O)CC(C(=O)NC(CF)C(F)(F)F)C(F)(F)C1 88592,C1(CC(=O)Nc2ccnnc2O)CCN(C(c2ccc(O)c(I)c2)=O)CC1O 88593,CC1=C(C(=O)NC(C2CCN(C(=O)COCc3cc(C)no3)C2)(C)C)SCCO1 88594,C1(C(=O)NCc2ccc(Cl)s2)C=CCN(C(C2CCCCO2)=O)C1 88595,C1(NC(COCCOC)=O)CC12CCN(C(=O)Cc1cnc(C)s1)C2 88596,C1(C)(NC(CC2C(C)CCN(C(C3CNC(=O)O3)=O)C2)=O)CC(C)(C)OC1=O 88597,C1(NC(CC(C)(C)C2CC2)=O)CCCN(C(c2ccc(Br)c(O)n2)=O)CC1 88598,Cc1cnccc1C(N1CCC(NC(=O)COC(c2nccn2C)C)C1)=O 88599,c1(C(N2C(CNC(Cc3ccc(OC)nc3)=O)CC2)=O)cc2n(n1)CC(F)C2 88600,C1(NC(c2cncnc2)=O)C(CC2CC2)CCN1C(=O)CCC1CC1 88601,C(=O)(CCC(F)(F)C(=O)N1CCN(C(C2C=C2C)=O)CC1COC)OCC 88602,Cc1cccc2c1OCC2C(=O)N1CC(CCCCNC(=O)CCOC(C)C)C1 88603,c1(CCNC(=O)NCCc2ccc(CC)cc2)ccc(OC)c(OC)c1OC 88604,C1(C(=O)NCCCCCCNC(C2(C)CC(C)C2)=O)Cc2ccncc2N1 88605,C(C(CC(C)C)NC(=O)Cc1ccc(C)cc1)NC(C1(NC(C)=O)CC1)=O 88606,C1(C(=O)NCC(C(C)(C)C)NC(C2ON=C(CC)C2)=O)Cc2cc(C)ccc2S1 88607,N1(Cc2cnc(CCC)s2)C(C(N2CCOC3(CC3)C2)=O)CC2CCCCC12 88608,c1(-n2cc(CC(C(=O)NC(C(CCCOC)C)=O)C)nn2)cccc(C#N)c1C 88609,C(C)(C(C(=O)Nc1cnn2ccccc12)C(C)C)NC(C1C(C(C)=O)C1(C)C)=O 88610,C(CC1CCCCC1)(C(=O)NCCCCCN(C(=O)C=Cc1cscn1)C)OC 88611,N1(C(C(CCOC)(C)C)=O)CCC2CC(NC(C3(O)CCSC3)=O)CCC2C1 88612,Cc1cn2c(n1)CC(C(=O)NCC(C(C)C)NC(c1cc(C3CC3)on1)=O)CC2 88613,C1(OCC(=O)NCC2(CC(=O)OC)CC2)CCN(C(C2(C)CCOC2)=O)C1 88614,c1(C(N2CCC(C)(NC(C(C)OCCOC)=O)C2)=O)[nH]c2ccc(Cl)cc2c1Cl 88615,CCC(C(=O)NC1(C(=O)OC)CC1)NC(=O)Cc1cn(C)nn1 88616,c1(C(N(CCOCCN(C(c2cn(CC=C)nn2)=O)C)C)=O)cc[n+]([O-])cc1 88617,c1(OC)ccc(Br)c(F)c1S(=O)(=O)N1CCC(N2CCCC2)C1C 88618,N1(C(C(C2CC2)NC(C(CC(C)(C)C)F)=O)=O)CC(C2CCCCC2)C1 88619,C(CC(=O)N1CCCCC1CCN(C)C(C1CCC(=O)O1)=O)(C(N)=O)NC(C)=O 88620,C1(CNC(C=C(COC)C)=O)CN(C(c2cccc(C#N)c2)=O)C2(CCC2)C1 88621,C1(CC)(NC(c2cc(CNC(C3CC(C)(C)C3)=O)on2)=O)CCCC1 88622,c1(C(=O)NC(CNC(CC(C)OC)=O)(C)Cn2cccn2)cccc(N)n1 88623,c1(SC)c(C(=O)NC(C(=O)NOCC(F)(F)F)C2CCOCC2)cnn1C 88624,C(=O)(C(CC=C)CC(C)C)NC1(CC=C)CCN(C(c2cccnn2)=O)CC1 88625,NS(=O)(=O)c1ccc(C(=O)NC2CN(C(=O)C(O)C(F)F)C2)cc1F 88626,CCC(C)(CNC(C1COCC(C)O1)=O)C(=O)N(C1CCN(C)C1)C 88627,c1(OC)ccc(NC(=O)CCC2CCN(C(C3CC3F)=O)CC2)cc1C 88628,N1(C(CCCCC=CCCC)=O)CCN(C(C2(C(F)F)CCCC2)=O)CC(O)C1 88629,Cc1cc(C(=O)NC2CC(F)(F)CC2NC(C2CCOC2C)=O)nc(O)n1 88630,C#CCC(CC(F)F)C(=O)NC(CC(C)C)C(=O)NCCNS(N)(=O)=O 88631,Cc1cc(C(=O)N(C)CC2(O)CCCN(C(C3CSCC(=O)N3)=O)C2)ncc1N 88632,C1(CNC(c2c(Cl)cn(CCC)n2)=O)CN(C(C2C(C#N)C2(C)C)=O)CC12CC2 88633,c1(C(N(CC)CC2CCCN2C(C2CC(CCO)C2)=O)=O)ccc(N(C)C)cn1 88634,C(=O)(CCCC(C)(C)NC(=O)COC1CCCOC1)NCC1(CC)CCC1 88635,N1(CC(=O)NCC(N(C(Cc2c(C)noc2)=O)C)C2CC2)CCN(C2CC2)C1=O 88636,N1(C(COC2CC(C(C)C)C2)=O)CC2(CC2)C1 88637,C1(CN(CCNC(c2ncccn2)=O)C2CC2)CC12CCOC2 88638,c1(OC)cc(F)c(CC(=O)N(CC(C)NC(c2csc3nccn23)=O)C)c(Cl)c1 88639,c1(C(N2CC3=C(C2)CN(C(=O)C(F)C2CCC2)C3)=O)ccn2cccc2c1 88640,N1(CCc2cn(C(C(N3CCC(O)(CC)C3)=O)C)nn2)C(C)CCCC1C 88641,C1(C(=O)NCc2cncc(CC)c2)CC12CCN(C(C1(O)CCCC1)=O)C2 88642,C1(CNC(CN(C)C(N)=O)=O)CN(C(=O)CC2C=CCCC2)CCC1(F)F 88643,Cc1cc(N(C)C(C2C3CN(C(C4CS(=O)C4)=O)CC23)=O)cc(C)c1 88644,N1(C(COCCC)=O)CCC2(CC1)CN(C(C1COCCO1)=O)C2 88645,C1(CNC(C2CCN(C)C2)=O)CCN(C(c2coc(C#N)c2)=O)CC1 88646,c1(C(=O)OC(C(=O)OC)C2CCCC2)cc(C(F)(F)F)nc2c1CCCC2 88647,C1(COC)(NC(c2cc(C(C)(F)F)on2)=O)CCN(C(C2CCC=CCC2)=O)C1 88648,C(=O)(CCC(F)(F)CN=[N+]=[N-])N(CCNC(C1CCc2nn[nH]c2C1)=O)CC 88649,n1(CCCSCC)nnnc1C(C(C)(C)C)NCC(C)C1CCC1 88650,c1(C(N2CCC(NC(c3ccc(O)nn3)=O)CC2)=O)cc2cc(F)ccc2o1 88651,C1(C)(N(C(C=CCN(C)CC)=O)C2CC2)CN(C(=O)CCCF)C1 88652,C(=O)(CC(C)CC(=O)N(C(C)C(=O)NCC(F)C1CCC1)C)OC 88653,c1(C(N(C(C)CCNC(=O)CCc2cncc(O)c2)C)=O)cccn2nncc12 88654,C1(CC(=O)NC2(CC=C)CC2)CCCC1NC(c1ccsn1)=O 88655,n1(CCNC(c2cn(CCNC(C(C)=C(CC)C)=O)nc2)=O)cccnc1=O 88656,c1(C(N2CCC(N(C(C3(C4CC4)CC3)=O)CC)C2)=O)cccn2c(C)nnc12 88657,N1(C(CC(C(CC)C)O)=O)CC2(CCN(C(=O)CC3CC(F)C3)CC2)C1 88658,Cc1cc(CNC(=O)NC2CCC(C(=O)O)C2)c(F)cc1Br 88659,c1(N(C)CC2(C(=O)NCC#N)CC2)ccc(C(C(=O)NC)OCC)c(C)n1 88660,CN1CC2(CC2)CC1C(N1CC(O)CC1C(=O)Nn1cccn1)=O 88661,S(=O)(=O)(C1CCS(=O)(=O)C1)NCC1CC(F)(CNC(=O)OC(C)(C)C)C1 88662,C(CCC(=O)NCC(O)C(=O)NCC1(SC)CC1)OCC 88663,N1(C(C=Cc2nc(C)sc2)=O)CCN(C(c2csc3nccn23)=O)CC(C)(F)C1 88664,C1(C(=O)Nc2n(C)nc(C3CC3)c2)CC(O)CCN1C(c1cncc(O)c1)=O 88665,N1(C(c2[nH]cc(C)n2)=O)CCCC(CCn2cc(C(C)O)nn2)CC1 88666,c1(CC)ccc(CCCNCc2nc(CO)n[nH]2)cc1 88667,N12CC(CC1(C)C)CC2=O.C(=O)(C(F)C(C)(F)F)NC1CC(N(C)CC)C1 88668,Cc1c(C(=O)N(CC(C)NC(c2ccc(C(F)F)cn2)=O)C)cnn1C(C)(C)C 88669,C1(NC(C(C(C)C)n2cccc2)=O)CN(C(c2nscc2Br)=O)CC12CC2 88670,C(=O)(CCCC(C)(C)C)NC1CN(C(Cc2ccc(C(=O)NC)cc2)=O)CC1C 88671,C(=O)(C1=CCCCC1)N1C(CO)CC(NC(C(c2ccc(F)cc2)C)=O)C1 88672,C(CC(C(=O)N1OC2CCC1C2)OC)NC(c1c(CC)cno1)=O 88673,C1(CNC(c2cccc(CC)c2)=O)CC2(CO1)CN(C(=O)C(C1CCC1)OC)C2 88674,c1(N(C)CC2COC(=O)O2)nc(N2CC3CC2C3)c2cnn(C)c2n1 88675,C1(NC(c2c(C)nn[nH]2)=O)CN(C(c2ccc(-c3ccc(Cl)cc3)[nH]2)=O)CC1C 88676,CC(C)C(CCNC(c1ccn(CCn2cccn2)n1)=O)NC(=O)CC(C)(C)O 88677,Cc1[nH]c(=N)ccc1C=CC(=O)NCCC(C)NC(C1CCCC12CC2)=O 88678,C1(CNC(C2CCC2(F)F)=O)CC2(CCN(C(c3cccc[n+]3[O-])=O)CC2)CO1 88679,C(=O)(C1=CCOC1)NC(C)CCCNC(c1cn(C2COC2)nn1)=O 88680,C12(C(N3CC(N(C)C)(C(N)=O)C3)=O)CCNCCCC1C2 88681,C#CCCCC(C)C(=O)N1CCN(C(c2cnoc2C)=O)CC1CCCC 88682,Cn1nc(Cn2cc(CN3CCCC(F)CC3)nn2)c2c1CCC2 88683,c1(OC)ccccc1OCCC(=O)NC1(CCNC(C2COCC(C)O2)=O)CC1 88684,c1(NC(C2(F)CCN(c3ncc(OCCOC)cn3)C2)=O)nc(C)c(Br)c(Cl)n1 88685,N1(C(C2C(C)C2)=O)CCCC(N(C(=O)CCC2CCCOC2)CCO)C1 88686,c1(C(=O)NCCCS(C)=O)ccc([N+](=O)[O-])cc1C(F)(F)F 88687,C1(C(N(C)CCC2CCCCN2C(c2cncc(Cl)c2)=O)=O)CCC(C)(C)CC1 88688,n1(CC(=O)OC)cccc(NC(C2CCC(O)(C(F)(F)F)CC2)=O)c1=O 88689,c1(CC(=O)NCC2N(C(C(N3CCC(O)CC3)C)=O)CC2)cccc(F)c1F 88690,CCCC(C)(CCC)C(=O)NCCC12CCC1CN(C(C1(C)CCSCC1)=O)C2 88691,C(c1ccsc1Br)=CC(=O)NC1CCC(CNC(c2ccoc2Cl)=O)C1 88692,N1(C(Cc2c(C(C)C)con2)=O)CCN(C(C)CNC(C2CCC(O)C2)=O)CC1 88693,N1(C(C(C(C)C)n2cncn2)=O)CCN(C(c2cncc(F)n2)=O)C2(CCC2)C1 88694,C(C(C)(O)CC(=O)NC1CCCN(C(c2cc(C#N)cs2)=O)C1)OC 88695,c1(NC(Cn2c(C)cc(C)n2)=O)ccc(NC(c2cnc(CO)cn2)=O)c(F)c1 88696,C=C(C)CN=C(NCCN1CCN(C(C)=O)CC1)NCC1CCC=CO1 88697,N1(C(c2cc(OC)ncc2)=O)CCN(C(C2CC(CCF)C2)=O)C(C2CC2)C1 88698,C(=O)(CC(CC)CC(F)(F)F)N1C(CN(C(CC(=O)NCC)=O)C)COCC1 88699,N1(C(CNC(c2n(C(C)C)ccc2)=O)=O)CCN(C(=O)CN(C)C(N)=O)CC1 88700,C12(C(N3CCCC(NC(CN(S(C)(=O)=O)C)=O)C3)=O)CCCN1S(=O)(=O)CC2 88701,C12(C(N3CC(NC(CSC(C)C)=O)C(CC4CC4)C3)=O)CCCCCC1OCC2 88702,C(CC(CC)C(=O)NC1CCCN(C(c2ncccc2C(F)F)=O)C1)=CC 88703,C(C(=O)N1CCC(C2CCCN2C(=O)CC2CC2)CC1)(C(C)C)SC 88704,C1(OC)(CNC(=O)COCC2CCCO2)CCN(C(c2ccccn2)=O)C1 88705,N1(C(CP(C)(C)=O)=O)CC2(CCCN(C(=O)Cc3cccc(C(F)F)c3)C2)C1 88706,C1(C(N(CC#CC)C(C)C)=O)C2CC3C(C2NC(=O)CC2CC(SC)C2)C13 88707,C1(F)(C(N2CCC(NC(c3cc(CN4CCOCC4)on3)=O)C2)=O)CC=CCC1 88708,c1(NC(c2cc(C)n(C(F)F)n2)=O)ncnc2ncc(Br)cc12.N1C(=S)NCC1 88709,N1(S(C)(=O)=O)CCCC(C2CCCN(C(c3cccc4c3C(=O)CCN4)=O)C2)C1 88710,Fc1ccc(CNC2(c3nnnn3CC3CC3)CCOCC2F)c(F)c1C(F)F 88711,Cc1ccc(NC(C2C(O)CCN2Cc2cc(F)c(O)c(Br)c2)=O)c(Cl)c1O 88712,CCC(CC)(c1nnnn1CCCC1CC1)NCC(C1CC1)C1CC1 88713,O=C(C1=C(F)CN(C(C2CN(C3COC3)C2)=O)CC1)NCC(F)CO 88714,n1(CCCC)nccc1C(=O)NC(C1CCN(C(=O)C(O)C2CC2)C1)C 88715,N1(C(C(N2CCN(CCF)CC2)=O)=O)CCCN2CCCC12 88716,c1(C(N(C(C)CNC(C2SCCS2)=O)CC)=O)ccc(C)o1 88717,C1(C(=O)NCc2nnc(N(C)C)s2)CN(C(=O)OC(C)(C)C)CCC1CO 88718,C(C(C)(C)CC(=O)NCC1CC(C(=O)NCC2OCCC2NC(N)=O)C1)N(C)C 88719,CC(C)(O)C(F)(F)C(=O)N1CC2(CC(C(=O)NC(CC3CC3)C3CC3)CO2)C1 88720,N1(C(c2cnn(CCC)c2Cl)=O)CCN(C(=O)C(F)n2cccn2)C(CCO)C1 88721,N1(C(C)C(=O)NCCCCNC(=O)CC(C)c2cnn(C)c2)CCC(O)CC1 88722,CCC(C)C(O)CC(=O)NCCN(C)C(c1ccn(-c2ccccc2OC)n1)=O 88723,CC1CCC(NC(=O)CCC2CC2)CN1C(c1cc(C2CC2)ccn1)=O 88724,c1(C(C(=O)NCC(n2cc(-c3cccnn3)nn2)C)(C)C)ccc(F)cc1 88725,C1(NC(Cc2nc(C)oc2)=O)CC2CCC(C1C)N2C(C1CN(S(C)(=O)=O)C1)=O 88726,Cc1ccc(CC(=O)NCC2CC3CN(C(C4CCCCC4O)=O)CC23)c(Cl)n1 88727,c1(CSC)ccc(C(=O)NC(c2ccccc2)CNC(c2n[nH]cc2CO)=O)o1 88728,N1(C(c2cn(CC)nc2)=O)CC(C2CC2)(C(=O)NC(c2cccc(C)n2)C)C1 88729,Cc1cc(C)c(C=CC(=O)N(CC(C)NC(c2cnc(Cl)[nH]2)=O)C)cc1C 88730,N1(CC(C)OC(=O)N(C)C)CCC2(CCN(C(=O)CC3CCC(=O)NC3=O)C2)CC1 88731,C1(CCC)CN(C(=O)CSC(C)(C)C)CCN1C(c1ncn(C(C)C)n1)=O 88732,C1(C(N2CC(NC(c3ccc(C(C)(C)C)[nH]3)=O)C2)=O)C2CCC(F)(F)C12 88733,c1(N(C)C)ccc(C(=O)NC2C=CC(CNC(=O)CCc3ncc[nH]3)C2)nn1 88734,N1(C(Cc2[nH]c(=N)sc2)=O)CC2CCN(C(=O)CC3CC4(C3)CC4F)CCC2C1 88735,N1(C(CCc2ccn(C)n2)=O)CCCC(C)(CNC(c2c(F)ccnc2F)=O)C1 88736,c1(-c2cccc(C(=O)NC(CCCOC)C(=O)NC)n2)ccc(C#N)c(C)c1 88737,c1(C(=O)NC2(CNC(CCSCC(C)C)=O)CCOC2)n[nH]c2c1NCCC2 88738,C12(SC)CC(C1)C(C)(C)O2.C1C(C)CC(=O)N1.c12cccc(c1)Sc1cn-2nn1 88739,CCCCC(CNC(=O)CC1(C)CC1(F)Cl)NC(c1scc(C)c1OC)=O 88740,c1(NC(N(C(C)C)Cc2cccc(C)c2)=O)cc(F)ncc1OC(=O)C(F)(F)F 88741,Cn1ccc(CC(=O)NCCCCNC(C2CCOC2)=O)n1 88742,C(=O)(C(CN=[N+]=[N-])NC(c1cc(Cl)n[nH]1)=O)NCCCN(C)C 88743,O=C1COc2ccc(F)cc2N1C(=O)N=c1cc(-c2ccccc2)o[nH]1 88744,CC1(C)CCCCC1CC(=O)NC1CC2CN(C(c3cc(C(N)=O)no3)=O)CC12 88745,N1(C(c2cnc(CC)nc2C)=O)CCC(CNC(=O)C(C)C(C)(C)C)C(F)(F)C1 88746,N1(C(CSC)=O)CCN(C(=O)CCOc2cccc3ccccc23)C(C)CC1C 88747,c1(C(=O)NC2(CNC(=O)CCc3cncc(F)c3)CC2)cc(O)cc([N+](=O)[O-])c1 88748,Cc1cc(-c2ccc(=NCc3ccc(CO)o3)[nH]n2)c(C)cc1-c1nn[nH]n1 88749,C1(NC(CCCOCC=C)=O)CCN(C(C2(C3CCCCO3)CC2)=O)CC1F 88750,C1(OC)CN(C(c2scnc2C(F)F)=O)CC1NC(=O)CCNC(N)=O 88751,C1(CCN(C(C2C(OC)C2C)=O)C(C2CCCC2)=O)CCC(C)(F)CC1 88752,N1(C(C2(OC)CCCCCC2)=O)CC(C)CN(C(=O)CCCCO)C(C)C1 88753,Cc1cc(CNC(=O)C(CNC(C2(C)CCNC2=O)=O)CC2CCCC2)sc1C 88754,C(N=c1[nH]c(Cl)nc2c1SCC2)C1CN(C(C2(C(N)=O)CC2)=O)C1 88755,C(N=c1[nH]cc(C#N)c2ccsc12)C1CCCC(NC(CCCC(=O)NC)=O)C1 88756,C1(CNC(C)=O)(COC)CCN(C(=O)Cn2ccc(C)n2)C1 88757,O=C(C1=CCC2CCC1N2C(C1CN2CCC1C2)=O)NCc1cccc(F)n1 88758,c1(C(=O)NCCC2N(C(COCCC)=O)CCC2)ccc(Cl)c(C)c1Cl 88759,C#CC1CCN(C(C2CCN(C(c3cn(C(C)C)nn3)=O)C2CC)=O)C1 88760,c1(C(N2CCOC(CCNC(C3(F)CC=CC3)=O)C2)=O)cccc(Br)c1 88761,N1(C(C(C)C#N)=O)CCC(C)(NC(=O)CCc2ccc(NS(C)(=O)=O)cc2)C1 88762,C1(CC(=O)NCC2(NC(C(CC)=CC)=O)CCC2)CCN(CC2CC2)CC1 88763,c1(C(CC)C)nccc(N(CC(O)CN(C(=O)CCOCC(F)(F)F)C)C)n1 88764,c1(C(N2CC(C(C)NC(c3c(C)scn3)=O)OCC2)=O)c(O)cccc1O 88765,C1(C(N2C(C)C(NC(=O)CC3(C)CCCCC3)CC2)=O)CC2CC1CC2O 88766,Cc1cc(CNc2ccc(-c3cc(O)ccc3F)s2)c(O)c(Br)c1 88767,C1(C(=O)NCc2csnn2)CC2(CCN1C(=O)CCC1CCCCC1)CC2 88768,N1(C(c2c(N)ccc(C(C)C)c2)=O)CCC2(CCC2)C(NC(c2cnsc2)=O)C1 88769,C12(NC(CCC(=O)NCC)=O)CCC(CC1NC(=O)CCn1ccnc1C)C2 88770,C=CC(CC)CC(=O)NCC1CC(OC)CN1C(C1CC1c1sccc1C)=O 88771,c1(C(=O)NC2CC(CNC(c3ccn(C)c3)=O)C2)cn(C)c(=O)c2ccccc12 88772,C(=O)(CC(C)CC(=O)NCC1(C)CCCN1C(c1cncc(OC)c1C)=O)OC 88773,C12(NC(C(C)SCC)=O)CCC(NC(c3ccnc(F)c3)=O)(CC1)C2 88774,S(=O)(=O)(CC(=O)N1CCN(c2ccc(F)cc2)CC1)NC(C)(C)C.C1CC(=O)N1 88775,c1(CC(=O)N(CCCNC(=O)CCN(S(C)(=O)=O)C)C(C)C)cncn1C 88776,c1(CC)ccc(C(=O)N(CCNC(C2CCN(C(=O)NC)C2)=O)C(C)C)c(F)c1 88777,C1(C(N(C)CCC2CCCO2)=O)(CO)CN(C(=O)CCOC2COC2)C1 88778,N1(C(c2cccc(C(N)=O)c2)C(=O)NCC)CCC2(CC1)OCC(C)(C)CO2 88779,c1(C(N2CCN(Cc3c(C)nc[nH]3)CC2CO)=O)cc(=O)c2ccccc2o1 88780,CCCC(C)C(=O)NC(C)CCCNC(c1cnn(CCN(C)C)c1C)=O 88781,CC(C(C)C(=O)NCc1cnc[nH]1)NC(=O)C=Cc1cnccn1 88782,c1(Cn2cc(CONC(CC3ON=C(C)C3)=O)nn2)ccc(F)cc1 88783,c1(C(=O)NCC(CNC(CNC(C(C)(C)C)=O)=O)CO)ccnc(O)c1F 88784,CC(CF)CC(=O)NC(C1CCN(C(c2[nH]nnc2-c2ccccc2)=O)CC1)C 88785,C(C#Cc1cnn(C)c1)NC(C1CC(NC(C(c2ccnn2C)C)=O)C(O)C1)=O 88786,Cc1cc(C#N)cnc1C(N1CCC(C(CO)NC(=O)CC2CC(C)C2)CC1)=O 88787,C1(F)(C(=O)NC2(CO)CC(C)C2)CCCN(C(=O)C(c2ccn(C)c2)C)C1 88788,c1(C(=O)NCC(C)NC(C(C)SCCCC)=O)ccc([N+](=O)[O-])cc1 88789,Cc1cn(C)nc1C(N1CCCC1C1CCN(C(c2cc[n+]([O-])cc2)=O)C1)=O 88790,C1(NC(CC(C=C)c2ccccc2)=O)(CO)CCCN(C(=O)C(C)C(O)CC)C1 88791,Cc1nn2c(C)c1C(=O)NC2.C1(Cc2ccccc2)CN(C(=O)C(N)=O)CC1C 88792,CC1(C)CC(O)CN1C(=O)NC1(c2ccccn2)CCC1 88793,C(=O)(C1=CCCN(C(=O)CNC(=O)CC(C)C)C1)NC(CC=C)C(=O)OC 88794,N1(C(C(C)S(C)(=O)=O)=O)C2CCC1C(F)C(NC(c1ccn3nccc3n1)=O)C2 88795,Cc1scnc1C(=O)NCCC(C)N(C)C(C1CSCCS1)=O 88796,c1(C(N2CC(C)CC(NC(C(C)SC)=O)C2)=O)c[nH]c2nccc(Cl)c12 88797,c1(C(N2CC(CNC(=O)C3=CCC3)C(F)(F)C2)=O)c(O)cc(=O)n2c1CCCC2 88798,N1(C(C(C)=C(CC)C)=O)CCC2CCN(C(c3ccc(Br)c(O)c3)=O)CC12 88799,CCC(C(=O)NCc1cc[nH]c1C(=O)NC(c1ccccn1)CO)NC(C)=O 88800,N1(C(C(Cc2cn(C(C)C)nn2)O)=O)CCC2(CCN2)CC1 88801,C(N=c1cc[nH]c(=NCCc2csc(C(C)(C)C)n2)[nH]1)c1cc(Br)cc(C)n1 88802,C(C(C)(O)C(=O)NCC1CN(C(=O)C(F)n2cccn2)CC1C)OC 88803,C(N=c1[nH]cnc(NCCOCCC(C)C)c1C)c1cn(CCC=C)nn1 88804,c1(CC)cc(C(=O)NCC2(O)CCN(C(c3cc(C4CC4)ns3)=O)C2)c(C)nn1 88805,c1(CN2CC(C)(C)C23CCC3)csc2ccc(F)cc12 88806,C(=O)(CCCN(C)N=O)N1CCN(C(CNC(CC(=O)OC)=O)C)CC1 88807,N1(C(CCCC(=O)c2cccc(OC)c2)=O)CCCn2nc(C#N)cc2C1 88808,N1(C(C=CC=CC)=O)CC2CCCC(NC(=O)Cn3cc(C#N)cn3)C2C1 88809,c1(CC(=O)N(CCC(C)NC(C2CCCOCC2)=O)C)nccc2ccccc12 88810,C(=O)(C1=NOC2(CCC2)C1)N(CCNC(C)=O)CCN(C)C.C(CO)S 88811,C1(C(=O)NCC2(C)CCN(C(CCc3cncc(C)c3)=O)C2)CN2CCC1CC2 88812,c1(C(N2CCC(OCCNC(c3cnc(CC)[nH]3)=O)C2)=O)nnccc1C 88813,C1(C(=O)NC2(CO)CN(C(C(C)=C(CC)C)=O)C2)CN2CCN1CC2C 88814,C1(N(C(c2c(C)ocn2)=O)C)CN(C(=O)CC2CCC(C)CO2)CC12CC2 88815,C1(CC)(CC)CC(C(=O)NC2CC(C)(NC(=O)Cc3cnc(C4CC4)[nH]3)C2)C1 88816,N1(C(C2CC(C#C)(O)C2)=O)CCOCC(C(=O)NCCC2CCCC3CC23)C1 88817,CC(C)CC(O)C(C)C(=O)NC(C)(C)CNC(c1nnn(C(C)(C)C)n1)=O 88818,C1(NC(c2c(C)cc[nH]2)=O)CCN(C(=O)Cn2ncc(Br)c2C)C(C)C1 88819,CC(C)CCC(O)C(=O)NCC1(C)CCCN1C(c1ccn(CC(C)C)n1)=O 88820,c1(CC)nc(C)c(C(=O)NCC2(NC(c3cnnn3C)=O)CC2)o1 88821,c1(C(N2CC(CNC(C(CCC)C)=O)C(C)C2)=O)cc(C)cc(Br)c1 88822,C12(C(=O)NCC3(CCNC(C(N4CCCC(O)C4)C)=O)CC3)CCOC(C)(C1)C2 88823,C(=O)(C(CC1CCCCC1)Sc1ccccc1)NCCC(=O)OC(C)(C)C 88824,c1(OC)ccc(OCCC(=O)NC(C)CCNC(=O)C(C#N)C2CC2)cc1 88825,C1(NC(c2cnc(CCC)s2)=O)CCC(C)(CNC(c2c(C)n[nH]c2C)=O)C1 88826,c1(C(N2C3CN(C(CSc4ccc(C)cc4)=O)C(C3)C2)=O)cnc2occc2c1 88827,CCC(O)C(C)C(=O)NC(c1cccc(OC)c1)CNC(c1ocnc1C)=O 88828,CC(C(=O)N1CCN(CC2CN(C(C3CC4(CC4)C3)=O)C2)CC1)C(F)(F)F 88829,N1(C(C(CSC)OC)=O)CCN(C(c2ccc(Cl)c(F)c2)=O)CC2(CC2)C1 88830,C(=O)(C1(C)CCc2ccccc21)NCC1(F)CCN(C(C(C#C)(C)C)=O)CC1 88831,c1(OC)ccc(F)c(C(=O)NC(C)CNC(=O)C=CC2CCOC2)c1 88832,N1(C(C2CCCCC2)C(=O)Nc2c(C)cccc2C)CCS(=O)CCC1C 88833,CC(C)(C(=O)NCC1CC1CNC(C1(C(F)F)CCCO1)=O)C1CCCO1 88834,CC1CC(CO)(NC(C2(F)CN(C(C3CCSC3)=O)C2)=O)C1 88835,Cc1cnn(C)c1CC(=O)NCC(O)CNC(=O)C(CN(C)C)N(C)C 88836,C1(C(=O)NCC(=O)NC2CC2)CC2CCC1N(C(=O)C=Cc1cnc[nH]1)C2 88837,C1(CC(=O)NCc2cc(C(N(C3CSC3)CC#C)=O)no2)CC(O)C1(C)C 88838,C=CC1CN(C(=O)CC2CCC2(C)C)CC1NC(c1ccc(OC)cc1F)=O 88839,C#Cc1cnc(C(=O)NC2CC(CCNC(=O)C=C(C3CC3)C3CC3)C2)c(C)c1 88840,Cc1c(NC(=O)NC2CC3(C2)CC(O)(C(F)(F)F)C3)cc(Br)cc1I 88841,c1(C(=O)NC2CCN(C(CCCCOC)=O)C2C)n[nH]c2ccc(OC)nc12 88842,Cc1ccc(C)c(CN2CCCC2CC(=O)NC(c2ccc(C#N)cc2)C)c1 88843,CC1CC(C)(C(=O)NC2COCC2NC(=O)Cn2cc(CO)nn2)CC(C)O1 88844,c1(OC)ccc(CC(=O)N(C)CCOCCNC(=O)C(F)C2CC2)c(C)c1 88845,CC(C)C(O)C(C)C(=O)N1CC2C(C(N3CCN(CCO)CC3)=O)C2C1 88846,C1(C(=O)NCC23CC(NC(CN4CCC(C)(C)C4)=O)(C2)C3)CC12CCCOC2 88847,C1(NC(=O)CCOC2CC2)CCC2(CC1)CC2NC(c1cc(C2CC2)ns1)=O 88848,NC(=O)CC(C(=O)NCC1C=CCCC1)NC(C1CC(C2CC2)C1)=O 88849,CC1=C(C(=O)N2CCC2CNC(C2CC2CF)=O)S(=O)(=O)CCO1 88850,C1(CNC(C(C)OCOC)=O)CC2CCC1N(C(=O)C(C)C(C)n1cccn1)C2 88851,CCC(C)C(O)CC(=O)NCC1CCCC1C(=O)NCC12CCC(CC1)CC2 88852,c1(C(N(CCCN(C(C2C(CC)CCCC2)=O)C)C)=O)cc(C)cc(C#N)c1 88853,CCCCCCCCC(C)CC(=O)N1CC(NC(=O)CS(=O)(=O)C2CC2)C(O)C1 88854,C1(C(N2CC(NC(CCSC)=O)C(CO)CC2)=O)C(C)(C)CCCC1(C)C 88855,C1(NC(CC(CC)(C)C)=O)CCCC2CN(C(C3(C(=O)OCC)CC3)=O)CC12 88856,n1(CC(=O)NC(CCC)CNC(c2ccnc(CC)c2)=O)cc([N+](=O)[O-])cn1 88857,N1(C(Cc2nc(C)[nH]n2)=O)CCC(NC(c2nc(C)nn2C)=O)C12CCC2 88858,C1(C(N2C(CNC(C3CC(C)(F)C3)=O)CC2)=O)CCN(c2ccncn2)CC1 88859,c1(C(=O)NCC2C(NC(c3c(CC)onc3C(F)(F)F)=O)C2)cc(C)cnc1N 88860,C(C(=O)N1CCC(O)(CNC(C2(c3ccccc3Cl)CCC2)=O)C1)(C(C)C)OC 88861,c1(CC(=O)NC2C(NC(CC(C=C)C)=O)COC2)ccc(Cl)c(Cl)c1 88862,c1(C(N2CC(CNC(C(CC#C)(C)C)=O)OCC2)=O)ccc2cc(C)ccc2n1 88863,c1(C(=O)NC2CCC(Nc3ncncc3Br)C2)ccc(C(F)(F)F)c(I)c1 88864,N1(C(c2ccn(C(CC)CC)n2)=O)CCC(C)(C)C1CNC(=O)Cc1ccncc1 88865,C1(NC(c2onc(C)c2C(F)(F)F)=O)CC(C)CN(C(=O)CCNC(=O)CO)C1 88866,N1(C(CCN(C)CC)=O)CCOC2(CCN(C(=O)C(C(C)C)n3ccnc3)C2)C1 88867,c1(COC)nc(NCC2C(C)CCCN2C(=O)C=CC(C)(C)SC)cc(O)n1 88868,CCC(F)(F)C(C)(C)C(=O)NC1CCC(CNC(c2cc(Cl)c[nH]2)=O)C1 88869,C1(C(N(CC(=O)N(C)C)C)=O)CCCC1CNC(=O)CCn1cccn1 88870,c1(C(N2CCC(NC(CC(C(C)C)C)=O)(CO)CC2)=O)cnn2c1CC(F)(F)C2 88871,C1(NC(CCC(C)O)=O)CCN(C(=O)CCCNC(N)=O)C(C)C1 88872,c1(C(N2CC(NC(C3CC=CCC3)=O)C(F)(F)C2)=O)cc(F)cc(F)c1F 88873,C1(CC(=O)NCC(C)CNC(C2CCCC2C)=O)Cc2ccccc2N1 88874,C(C(=O)N=S(=O)(c1ccc(Br)cc1)C(F)F)n1ccc(C)n1 88875,c1(C(N2CCCC(F)(CNC(C(C)(C)F)=O)C2)=O)cn2cccc(Br)c2n1 88876,C1(NC(C(N2CC3OCC(OC)C3C2)=O)=O)C2CC3CC1CC(O)(C3)C2 88877,C1(CN(C)C(C2CC(CF)C2)=O)CCCCN1C(C12CCC(C1)C2)=O 88878,N1(C(c2c(C)ncnc2)=O)CCC(C(F)(F)F)C(CNC(=O)CC2CCCO2)C1 88879,Cc1cnc2cccc(C(=O)NCC3CCN3C(=O)C=Cc3cc[nH]c3)n12 88880,C1(C(=O)NCCC(COC)OC)CN(C(=O)CC2CC=CC2)C(C)(C)C1 88881,Cc1csc(=NCC(=O)NCC2COCC2NC(c2c[nH]cc2C(C)(C)C)=O)[nH]1 88882,CCCC(CC)CCC(=O)NCC(C)CC(=O)NC1CCN(CCOC)C1 88883,C1(NC(C2C(C(=O)OCC)C2)=O)CCN(C(=O)Cc2cnn(C)c2C)C12CCC2 88884,C(=O)(C1=CCCC1P(C)(C)=O)NC1(C)CN(C(c2ncncc2Cl)=O)C1 88885,N1(C(COCC#C)=O)CCC2(CCC2)C(NC(=O)C(C)CC(C)(C)C)C1 88886,C(CCS(=O)(=O)c1ccc(F)cc1)N1c2c(cc(F)cc2)CC(CCC(=O)O)C1 88887,N1(C(C(CC)F)=O)CCC(O)(CN(C)C(C2CCCCN2C(=O)C(C)C)=O)CC1 88888,Cc1cc(C(N2CCC(C)N(C(C3SCCC3C)=O)CC2)=O)c(C)cc1Br 88889,C(C(F)(C(=O)NCC1(C#N)CC1)C(C)C)NC(c1c(C)scn1)=O 88890,C(=O)(C1=NOC(C)(C)C1)N1C(CN(C(c2cnc3n2CCC3)=O)CC)CCCC1 88891,CN1CC(O)CC1C(=O)NCCCNC(=O)C(C)(C)N1CCCC1 88892,C(CO)(CCCCNC(=O)CCN1C(=O)CCC1=O)NC(C(C)(C)C1CC1)=O 88893,c1(NC(C(C)C(=O)NCC(=O)OC(C)(C)C)C)cccc2cncn12 88894,c1(OC)cccc(Cl)c1CNC(=O)C(=O)NCC(c1ccc(Cl)c(Cl)c1)N(C)C 88895,Cc1c(C(=O)N(CC(O)CNC(c2ccc(CF)cc2)=O)C)oc2ccccc12 88896,c1(C(=O)NC2C(C)CN(C(c3ncc(F)cn3)=O)CC2)cccc2c1ncn2C 88897,N1(C(C2COCCN(C(c3ccns3)=O)C2)=O)Cc2ccncc2C1 88898,c1(C(N2C3(CNC(=O)C(F)CC4CCCC4)CC(C2)C3)=O)cc2occc2s1 88899,C(CNC(=O)C=CC(F)(F)F)(C(C)C(C)C)NC(C(c1cc(C)sc1)(F)F)=O 88900,N1(CCCC(=O)NCCNC(c2c(C(C)(C)C)con2)=O)C(=O)CNC1=O 88901,N1(C(c2c(CC)cns2)=O)CC(C(=O)NCC2CC23CCOCC3)CC(C)C1 88902,N1(c2nc(N3CCC4CCC(C3)S4)cc(C)n2)CC2CC3CC(C2)CC1C3 88903,Cc1cocc1C(=O)NCC(O)CCNC(=O)C(C)CF 88904,N1(C(CCCOCCC)=O)CC2(CCC2NC(c2ccc(F)cc2CC)=O)C1 88905,CC(CN=c1ncc2ccccc2[nH]1)N(C(=O)C1=CC2CCCC12)C 88906,c1(C(N2CC(OC)C(F)C2)=O)cnc2c(-c3ccc(I)cc3)cnn2c1 88907,c1(C(N(CC(C)O)CCNC(=O)Cc2cc[nH]n2)=O)cccc2c1OCC(=O)N2 88908,C1(CNC(C(C2CCCCC2)OC)=O)CN(C(C2C=CC=CC=C2)=O)CCN1C 88909,C1(CNC(C(C)(C)C2CCOCC2)=O)CCCCN(C(=O)C(F)OC(F)(F)F)C1 88910,c1(CNC2C(C(N(C3CCOCC3)CC)=O)CCC2)ccc2ccc(Cl)cc2n1 88911,C1(N(C(Cc2c(C)cccn2)=O)C)CN(C(C2CC3CCC2CC3)=O)CCC1C 88912,N1(C(c2cc(OC)ns2)=O)CCCC(N(C(=O)CN2CCC2C)CCF)C1 88913,C1(C)(OC)CC(NC(c2ccc(CNC(=O)C(C)NC=O)nc2)=O)C1(C)C 88914,C(C(CO)C(C)(C)C)NC(CC1N(C(C2CC(N(C)C)C2)=O)CC1)=O 88915,c1(N(C(C2CCC(C(C)C)C2)=O)CC2CCN(C)CC2)ccc(F)c(F)c1 88916,C=C=CCCN=c1[nH]c(N2CCC(C)(CN(C)C)C2)nc2c1COCC2 88917,C1(CC(=O)NCC2(C(N3CC(n4cnnc4)C3)=O)CCCC2)COCC1O 88918,N1(C(c2c(CC)occ2)=O)CC2CCC1C(NC(=O)CCCC(N)=O)C2 88919,C(=O)(C(F)CC(C)(C)NC(=O)CC#N)NC(C(C(C)C)O)C 88920,c1(C(=O)NC2CC(NC(C(COC)(C)C)=O)C2)cc(OC(F)F)cc(F)c1 88921,N1(C(CC(C)N(C(c2cncc(C)c2)=O)C)=O)CC(C(C)C)CCC1C 88922,C(CN=c1[nH]c(=NCC2(F)CCC2)c2[nH]ccc2[nH]1)NC(=O)NCC(C)C 88923,C1(CCOC)(NC(COCC(=C)C)=O)CCN(C(=O)C(CCSC)NC=O)C1 88924,C1(CNC(C2CC=CCO2)=O)C2CN(C(=O)CN3CC=CC3)CC12 88925,Cn1ncc2c(=O)n(Cc3nccn3-c3cccc(F)c3)cnc12 88926,C(C)(CC(C)(C)C#N)(c1n(C)nnn1)NC(C)CCCCCCO 88927,c1(CC(N2C(CNC(CCCC#CC)=O)COCC2)=O)c[nH]c2cccc(C)c12 88928,c1(-n2cc(C(=O)OCC)nn2)cccc(C(N2CCOC(C(=O)N(C)C)C2)=O)c1 88929,C(c1ccccc1)=CC(=O)NCCOCC(=O)NCCCCN(C)C 88930,C1(C(N2CCCN(C(=O)Cc3cccc(Cl)c3Cl)CC2)=O)CCCC12OCCO2 88931,Cc1nc2cc(NC(C3CC(O)CN3C(c3ccn(C)c3)=O)=O)ccc2s1 88932,c1(SC)ccccc1CC(=O)NC1CC(=O)N(C2CN(C(c3ccns3)=O)C2)C1 88933,n1(COC)nccc1C(=O)NC(C)CC(C)NC(=O)CC1CCCC1 88934,Cc1n[nH]c(C)c1C(C)NC(=O)C(CNC(=O)OC(C)(C)C)CC1CCCCC1 88935,CC1CCc2[nH]nc(C(=O)NC(C3CCCN3C(c3cc(O)n(C)n3)=O)C)c2C1 88936,C12(NC(C3N(C)CCCC3)=O)CCC(C(=O)NCC3CCC(O)CC3)(CC1)C2 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89060,n1(CCC(=O)NCC2N(C(C3N(C(C)(C)C)CC3)=O)CC2)cc(Br)cn1 89061,C(C(C)(C)C(=O)NCC1(C2CCC2)CC1)N(C)C.C12CCCC1NC2=O 89062,CC(C)CC(C)(C)C(=O)NCC1CCCN1C(C12CC(CO1)C2)=O 89063,c1(N2CCC(N(C(=O)C(=O)NCc3ccc(F)cc3)CC)C2)nc(C)nc(C)c1F 89064,C(=O)(CCC(C)(C)c1ccccc1)NC(C(C)C)C(C)NC(=O)Cc1cn[nH]c1 89065,C(C)(N=c1[nH]c(N2CCOC(C(N)=O)C2)nc(=N)[nH]1)c1scc(C)n1 89066,C1(NC(CCSCCCC)=O)CCCC(CN(C)C(C2COC2)=O)C1 89067,C(=O)(C(COC)CC(C)C)N(CCC)CCNC(C1CCCCC1(F)F)=O 89068,C(c1ccc(OCCF)cc1)=CC(=O)NCC(C1CC1)NC(C12CCC1CC2)=O 89069,c1(C(N2CCC(CNC(c3n[nH]c4ncccc34)=O)C2)=O)c(F)ccc(O)c1F 89070,C12(C(=O)NCCCOCCNC(C(n3cc(C)nc3)(C)C)=O)CCCCC1C2 89071,C1(C(N2CCCC(C)(OC)C2)=O)(OC)CCC(C)(C)C1.C12CCCCC1C(=O)N2 89072,C1(NC(=O)CC2CC2)CCOC12CCN(C(c1csc3c(Cl)cccc13)=O)CC2 89073,c1(CCNC(N(CC(C)(C)C)C2CCCC2)=O)nc(C(F)(F)F)cs1 89074,C(CCC(=O)NC(C1CN(C(C2CNC(=O)O2)=O)C1)CO)OC(C)(C)C 89075,Fc1cc(NC(CCc2cn[nH]c2)C(F)F)cc(CC2CCCO2)c1 89076,C(=O)(C1CCCn2ncnc21)N1CCN(C(CNC(=O)NC)=O)C(CCOC)C1 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89094,C1(NC(C)=O)CCN(c2ncco2)CC1.C12CCCN(C1)C(C)(C)c1cn2nn1 89095,C1(NC(COCC(=O)NC)=O)COC2(C1)CN(C(=O)C(C(C)C)OCC)C2 89096,C1(C(=O)NCCCC#C)C2CCC(C2)C1NC(C1(CO)CCOCC1)=O 89097,C1(NC(C=CCC)=O)CN(C(c2cc(OCC)no2)=O)C(C)(COC)C1 89098,CC1(C)CN(C(=O)C=Cc2ccc([N+](=O)[O-])s2)CCN(C(C2(C)CC2(F)F)=O)C1 89099,C(=O)(Nn1cnnc1)C1C(C)(C)C1N(C(=O)CC12CCCC1C2)CCO 89100,CC12CCC(C(=O)NC3CCCC(NC(C45CC6CC4C5C6O)=O)C3)(CO1)C2 89101,c1(NC(N)=O)cc2n(n1)CC(Nc1cnc(CNC(=O)OC(C)(C)C)nc1)CO2 89102,C1(c2ccc(Br)cc2)(NC(C2CCS2)=O)CCCCC1 89103,Cc1cc(C(=O)NC2CC(O)CN(C(c3cc(C(N)=O)co3)=O)C2)ncc1F 89104,Cc1cc(N)c(C(N2CCN(C(C3CCCS3)=O)CC2C(C)C)=O)cc1C 89105,C(=O)(C1CCCc2ccccc21)N1CC(C)N(C(c2cccc(O)n2)=O)CCC1 89106,C1(NC(C(C(=O)OC)C)=O)CN(C(=O)CCN2CCCS2(=O)=O)CC12CC2 89107,N1(C(CCC=CC)=O)Cc2ccccc2C1C(=O)Nc1cncc(C(F)F)c1 89108,N1(C(C(CC#C)O)=O)CC2CCC1CN2C(=O)C(C(C)(C)C)SC 89109,c1(-c2nc(C(=O)NCCC3(CSC)CC3)sc2)cccc(C#N)c1 89110,c1(NCC(N2CCC(C(C)NC(CN3CC(C)C3)=O)C2)=O)ccc(O)cc1 89111,C1(CNC(c2c(CC)ncnc2)=O)(NC(=O)C(C)NC(=O)NC)CCCCC1C 89112,c1(N2C(C)(CNC(C(C)(C)O)=O)CCC2)nc2c(F)cc(Cl)cc2s1 89113,CCC(C#N)C(=O)NC(CCSC)C(=O)N(CC1CC1)CC1CC1 89114,c1(C(=O)NC2(CC=C)CN(C(C3(c4cc[nH]n4)CC3)=O)C2)cccc(C(N)=O)c1 89115,C(=O)(C(CC)CC(C)C)NCC1C(NC(CN(CCC#C)C)=O)C1 89116,CN1CC(C(=O)NC(CC2CCC2)C(=O)NCC2(C(C)(F)F)CC2)CCC1=O 89117,c1(C(=O)NCCN(CC(C)O)C(C2CCC2)=O)cc2sc(Br)cc2[nH]1 89118,N1(C(CCc2cc(OC)no2)=O)CC(CNC(=O)C(C)N2CCC2)C(C)C1 89119,C1(NC(CC2C(C)C2)=O)CC2(C1)CC(NC(c1ncoc1C1CC1)=O)C2 89120,C1(CC(=O)NCC2(NC(=O)COCC3CCCOC3)CCOC2)CC2(CC2)C1 89121,c1(C(N(CC(O)CN(C)C(c2cn(-c3nccs3)nn2)=O)C)=O)csc(C#N)c1 89122,O=C(CC1=CCCCC1)NCCOC1CCN(C(=O)CCCn2cccn2)C1 89123,Cn1cc(Cl)c(C(=O)NC2CC3(C2)CC3C(N2CCCC(F)C2)=O)n1 89124,c1(NC2(CN(C(CCOCC(=O)OCC=C)=O)C)CC2)ccc(C(C)=O)c(F)c1 89125,C1(CC(N2CC(OCC(C)C)C2)=O)C2CCCC2N1C(=O)C(C)(C)CN(C)C 89126,C12(CNC(C(C)N(C(=O)Cn3ccnc3C)CCC)=O)CCCC(CO1)C2 89127,C(=O)(N=c1cc(Cl)cn[nH]1)C1C(NC(c2cc(C)ncc2)=O)C1 89128,N1(C(c2ccc(SC)cc2)=O)CC2(C)CC1C2CNC(=O)Cc1ccc(C)nc1 89129,c1(OCC)cc(N2CCC(C(C)NC(=O)C(C)(C)O)C2)ncn1 89130,C1(C(=O)NCC2(CSC)CC2)C2CN(C(=O)CC3CC4CC4C3)CC12 89131,C(=O)(C(C)(N)C(F)(F)F)NCc1n(CC)nnc1C 89132,N1(C(C(C)n2cnnn2)=O)CC2(C1)CN(C(c1c[nH]cc1C1CC1)=O)CCO2 89133,C1(CNC(C(C)C2CCOC2)=O)(CNC(C2(C)COC2)=O)CC1(F)F 89134,c1(C(=O)NC2C(NC(C=C(C)C(C)(C)C)=O)C2)oc(Br)nc1C 89135,C1(C(N2CCCN(C(CC3CCC(C)CC3)=O)CC2)=O)CCCCN(C)C1=O 89136,CS(=O)C=CC(=O)NC1(CNC(=O)Cn2cc(I)nn2)CC1 89137,C1(C#N)(CC(N2CC(C(C)NC(=O)NCCCl)C2)=O)CCOCC1 89138,N1(C(COCC(C)C)=O)CCC(O)(CN(C)C(C2CCCN2C(C)C)=O)C1 89139,c1(C(N2CCC(NC(C(CCC)=CCC)=O)(CO)C2)=O)cc2ncccc2[nH]1 89140,C1(C)(CC)CC(NC(c2c[nH]nc2OC)=O)CN1C(=O)Cc1ccnn1C 89141,C1(C(=O)NCC2(CNC(c3c(N(C)C)ccnc3)=O)CCC2)CCCCNC1=O 89142,c12cncc(c1)C(=O)NC1CC(C1)CO2.C1(CC)CC(n2ccnn2)C1 89143,C1(CNC(C2C(C)C2)=O)CC2(CO1)CN(C(=O)CNC(=O)C1CC1)C2 89144,N1(C(C(CC2CCC2)OC)=O)CC2CC(C1)N2C(=O)Cc1ccc(Cl)cc1 89145,c1(C(=O)NCc2nc(CNC(CC(C)(C)O)=O)sc2)cc(O)nc(C2CC2)n1 89146,c1(NCC)ccc(F)c(C(=O)NCCN(C(=O)C(CC)NC(N)=O)CC(C)O)c1 89147,CCC(C)(CCC(C)C)C(=O)N1CC2CN(Cc3c(OC)cccc3Cl)C2C1 89148,C1(NC(C(C)OCC#C)=O)CCC(N(C(=O)C(F)CC2CCCCC2)C)CC1 89149,c1(C(=O)NC(CCCCC#C)=O)ccc2c(c1)CN(C(C1CCN(CC)C1)=O)C2 89150,c1(C(=O)NC2CC(C)(NC(C(C)NC(=O)OC)=O)C2)cccc(OCC(F)F)c1 89151,CC(CC(=O)NCC(O)CNC(=O)CS(=O)(=O)CC1CCCO1)C(F)(F)F 89152,n1(CC)c(C(=O)N(C(c2ccccc2)CNC(C2(F)CC2C)=O)C)cnc1O 89153,C#CCC(CC(=O)Nc1cc(OC)cc(Cl)c1)NC(C1CCN(C)C1)=O 89154,CN1Cc2cc(NC(=O)NC3CCc4ncnn4C3)ccc2C1=O 89155,C(=O)(CCN=C(NCC1CCN(S(C)(=O)=O)C1)NC1CCOCC1F)NC 89156,c1(CC)nc(C(N2CC(NC(=O)C(C)NC(c3ccco3)=O)C2)=O)cs1 89157,c1(-c2nc(C3CCC(C)CC3)nn2C(C2CCOCC2)C)nccc2occc12 89158,C1(CNC(CC(=O)NCC#C)=O)CCCN(C(C2CC(C)CCO2)=O)CC1 89159,C1(C(=O)NCC(CC)NC(c2n[nH]cc2C2CCC2)=O)CCC(C)CC1 89160,c1(OC(C(=O)NCC(CCNC(C2CC(C)(F)C2)=O)O)(C)C)c(F)cccc1F 89161,N1(C(C(C=CC)O)=O)CCCC12CCN(C(C1CC(=O)CCO1)=O)C2 89162,c1(C(=O)NC23CN(C(Cn4c(C)cc(C(F)F)n4)=O)C(C2)C3)ccc(F)c(F)c1 89163,S(=O)(=O)(c1ccc(NCC2(C)CCC(=O)N2)c(F)c1)N1CCC(CC=C)C1 89164,C1(C(=O)NCc2ccc(C)s2)CC(N=[N+]=[N-])CN1C(=O)C(F)C1CCC1 89165,C#CC1(NC(C2(C)CCN(C(=O)C(C)SC(C)C)C2)=O)CCOC1 89166,N1(C(C(=O)NCc2csc(C(=O)C3CC3)c2)=O)CC(O)CC(F)C1 89167,CC1(C)CC(C(=O)NC2CCCCN(C(c3c[nH]nc3C(F)(F)F)=O)C2)=NO1 89168,C1(COC)CN(C(=O)C(c2cc(C)cc(F)c2)C)CCN1C(c1occc1C)=O 89169,Cc1cc(C(=O)NCC2CN(C(c3cnncc3C(F)(F)F)=O)C2)cc(N)c1O 89170,Cc1n[nH]cc1C(=O)NC1CC(CCNC(=O)CCSc2nccn2C)C1 89171,CCCCC(CNC(=O)CCOCc1ccccc1)NC(=O)C(O)CC 89172,c1(C(=O)NC(C)C)n[nH]cc1C(=O)NC1CC(N(C(=O)CC2CCOC2C)C)C1 89173,C1(CNC(C(C(CC)O)C)=O)CCC2CN(C(c3nc(C)sc3C)=O)CC12 89174,C#Cc1cccc(C(=O)NCC2CN(C(=O)Cn3cc([N+](=O)[O-])cn3)C2)c1F 89175,N1(C(=O)NC)CCCC(C(=O)NCC2(OC)CN(C(=O)C(C3CC3)OC)C2)C1 89176,C(CCC(=O)NC(Cc1ccccc1)CCNC(=O)COC1CCOC1)OCC 89177,CC(C)(CCF)C(=O)NC1CC(O)(CNC(C2CC(CC3CC3)C2)=O)C1 89178,c1(N2CCOCC(NC(C(c3cccnc3)OC)=O)C2)ccn2ccnc2n1 89179,N1(C(c2nc(CCC)oc2)=O)CC(NC(c2cnc(C3CC3)s2)=O)C(O)C1 89180,O=C1OC2CC1N(C(=O)CCC1CCCCO1)C2 89181,c1(CC)nc(CNC(C2(NC(C3CC(=O)CS3)=O)CC(O)C2)=O)n[nH]1 89182,C1(C(N2CCC(SC)CC2)=O)CCC2CCCC12.C12CCC(C1)n1cc(nn1)C2N 89183,C(CC1=CCN(C(C2CCc3ccnn3C2)=O)CC1)NC(C(C)(O)C1CC1)=O 89184,C(=O)(CCC(=O)NN(C)C)N1CC(C)N(C(=O)CNc2cccnc2)CC1 89185,c1(C(=O)OC)ccc(F)c(C(N2CCN(C(c3cc(Cl)c[nH]3)=O)CC2CF)=O)c1 89186,c1(C(=O)NC2CC(NC(C3C4CC5C(C4=O)C35)=O)C2)ccc2c(n1)CCO2 89187,Cc1c(C(=O)NC(CN(CCO)C(C)C)C2CCC2)cccc1Cl 89188,c1(C(=O)NCCCCNC(C=C(CC)C)=O)cc(C)n(C)c(=O)c1 89189,N1(C(CC=C(C)C)=O)CCOC(CNC(=O)CC23COCC(C2)C3)C1 89190,Cc1cc(C)c(C(N2CC(N3CCN(C(C4CC(F)C4)=O)CC3)C2)=O)[nH]1 89191,N1(C(CSc2nc(C)[nH]n2)=O)C(CNC(C2(n3cnnn3)CC2)=O)CC2COCC12 89192,C(=O)(CC(C)C(F)(F)F)NC(CCN(C(CCCCOC)=O)C)C 89193,C1(O)(C(=O)NC2CC(C(N3C(C)(C(=O)OCC)CCC3)=O)C2)CCOC1(C)C 89194,Cn1c(C(N2CC(CNC(C3CC(C)(C)CO3)=O)C2)=O)cc2sccc12 89195,C(=O)(C(CCNC(C1C2CCCOC12)=O)OC)NCCC1(COC)CCC1 89196,c1(OC)nc(C)ccc1C(=O)N(CCCn1cc(C2(OC)COC2)nn1)C 89197,N1(C(c2c(C)nn(C(C)C)c2)=O)CC(NC(=O)CC=C(Cl)Cl)CCC1C 89198,C(c1c[nH]c2ccccc12)=CC(N1C(C(N2C(C)C(O)CCC2)=O)CC(O)C1)=O 89199,C1(CC(=O)N(CC#C)CC=C)CCN(C(=O)C(C)C2CCC2)C1(C)C 89200,c1(C(C)C(=O)NCCOC(C2(CC(=O)N(C)C)CC2)=O)cnn(C)c1 89201,C(=O)(C(C)(CC)OC)N1CC(CC=C)(C(=O)NCC2(COC)CC2)C1 89202,C1(NC(Cc2c(CC)cccc2)=O)CC2(C1)CN(C(=O)Cn1cnnc1O)C2 89203,N1(C(c2c(C)ncn2C)=O)CCC2(CCCN2C(c2cncc(Cl)n2)=O)C1 89204,CC1CN(C(=O)COCC2CC2)CC(C)C1NC(=O)CCCN(C)N=O 89205,C1(C(N2CCC(CCNC(C3(CO)CC(F)(F)C3)=O)C2)=O)CC2CCCC(C1)C2 89206,c1(C(N(CCC)CCNC(c2sccc2Cl)=O)=O)ccc(F)c(C)c1C#N 89207,c1(NC(CCC)C)ncnc(NCCc2ncccc2C)c1C 89208,Cc1ncc(C(=O)NCC2CCCCN(C(c3cncs3)=O)C2)cc1N 89209,c1(C(=O)NC(CC)CN(C)C(C2CCCO2)=O)c[nH]c2c(Cl)cccc12 89210,N1(C(C2ON=C(C(=O)OC)C2)=O)CCOCC(C)(CNC(c2cnc(Cl)[nH]2)=O)C1 89211,S(=O)(=O)(c1cccc(C)c1)N1CCC(C(=O)NCCCCCN(C)CC)C(O)C1 89212,C1(C(=O)NCC(CO)NC(C2(C=C)CCCCC2)=O)CNC(=O)CC12CCC2 89213,C1(NC(c2cnc(COC)s2)=O)CC2CC1CN2C(c1cn(C)c(C)n1)=O 89214,Cc1csc2ncc(C(=O)N(C)CC3CC(F)CN3C(=O)CC3(C)CC3)n12 89215,C=Cc1cnn(C)c1C(=O)NCC1CN(C(=O)C(F)(F)CC)CC1C(F)(F)F 89216,Cc1cc2c(C(N3CCSCC3CCNC(C34CC(C)C3C4)=O)=O)cccc2o1 89217,c1(NCC2CCCN(C(C)=O)C2)[nH]c(=NCCCC2CCC2)nc2c1ncn2C 89218,Cc1nc(C)n(CCC(=O)NCC2(C(C)(C)O)CN(C(=O)CC(F)(F)F)C2)n1 89219,N1(C(c2c(CC)oc(C)c2)=O)CC2CCCC(C1)N2C(C1CC2(C1)CC(F)C2)=O 89220,n1(CCNC(=O)C(C)CC(N)=O)nnc2c(N3CCC(=CCOC)CC3)ncnc12 89221,N1(C(C(COCC)(C)C)=O)CC2(CNC(=O)CC(C)(O)C3CC3)CC1(COC)C2 89222,C1(C(=O)NCC2(F)CC(NC(C3(CF)COC3)=O)C2)CCCCCC1 89223,c1(NC(C2(OC)CCN(C(C(CCCOC)C)=O)C2)=O)cn(C)c(=O)nc1O 89224,C1(C(C)NC(=O)CCCN(C)C)CCN(C(c2c[nH]c(=S)cn2)=O)CC1 89225,N1(C(=O)C(F)F)CCCC2C1CCN2C(c1ccc(OC(F)(F)F)c(F)c1)=O 89226,C(CCCC(=O)NC1(CN(C)C(C2(CCO)CC2)=O)CC1)OCC 89227,C1(NCCn2cnc(C)c2C)CCC2COCCC2(C#N)C1 89228,CC1(C)CC(C(=O)NC2CCC2NC(=O)Cc2ccc(Cl)cc2)C(C)(C)O1 89229,CC(C)C(CNC(=O)CP(C)(C)=O)C(=O)NC(C)(CO)C(C)(C)O 89230,c1(CC)nn(C)c(Cl)c1C(N1CCC(O)(CNC(=O)C(F)(F)CN(C)C)C1)=O 89231,CC12CC(C(=O)NCC(O)CCNC(=O)C(O)CN3CCCC3)(CCO1)C2 89232,c1(-c2cn(CCN3CCC(C)CC3)nn2)ccc(Cl)cc1F.C1CC(=O)N2CCC12 89233,C(C)(C)(CCC(=O)N(C)CC1CN(C(=O)C(c2ccc(Cl)s2)C)CCO1)OC 89234,c1(OC)cc(CNC(=O)CC2(C)CN(Cc3cc(CO)ccc3O)C2)ccc1F 89235,c1(C(=O)NCC2C3CN(C(=O)CC4CC=CCC4)CC23)cc(O)ncn1 89236,Nc1cc(Cl)cc(Cl)c1C(=O)NCCC(O)CNC(c1cnc(C2CC2)[nH]1)=O 89237,c1(C(N2CCC(CNC(c3c(C)n(C)nc3)=O)C2)=O)cc(Br)cc2nc[nH]c12 89238,c1(SC)ccc(C(=O)NCC2(F)CC(CNC(=O)C=CC3CCCO3)C2)o1 89239,c1(C(N(CC2(NC(CN(CCC#C)C)=O)CC2)CC)=O)cnnc(O)c1 89240,C(=O)(CCCCN(C)C)NCC1CC(C)(NC(c2[nH]cc(C(C)=O)c2)=O)C1 89241,C1(C(=O)NC2CC3COCC3C2)C2CC(C(O)C2O)S1(=O)=O 89242,CCC(C)N(OC)C(=O)C1CC(=O)CN1C(C1CC2(C1)CC2(F)F)=O 89243,c1(C(C)C)nccn1CC(=O)NCC(O)CN(C)C(C1CC1C(C)(C)C)=O 89244,CC(C)C(C)C(CNC(=O)Cc1c(Cl)cnn1C)NC(=O)COCC1CCC1 89245,C(C(=O)Nn1nnc(C)c1C)(C1CCCC1)N(C(C(NOC)=O)=O)C1CC1 89246,CC(C)C(C)(CNC(=O)C(C)Oc1ccc(F)cc1)NC(=O)C=Cc1cocn1 89247,N1(C(c2nc(C(c3ccccc3)C)sc2)=O)CC(C(=O)O)CCC1C(=O)O 89248,Cc1cccc(CCCNC(c2nc[nH]n2)C)c1 89249,c1(C(=O)NCCC2CCCCN2C(=O)C(F)C2CCOC2)ccc2ocnc2c1 89250,c1(C(=O)NC2CCN(C(CCC(=O)OCC)=O)CC2C)cnc2n[nH]c(C)c2c1 89251,c1(OCCC)ccc(C#CCN=c2cc[nH]c(C)c2)cc1 89252,C1(S(N)(=O)=O)(C(=O)NC(C(C)NC(C2CCCC(=O)N2)=O)CO)CCC1 89253,C(=O)(CC(O)CC(C)(C)C)N1CCC(CN(C(CCCn2ncc(C)c2)=O)C)C1 89254,c1(OC)ccc(O)c(NC(=O)C(C)=CCNC(=O)CCCCCSC)c1 89255,C1(CC)CN(C(c2occc2CNC(=O)C(n2cc(C)cn2)C)=O)CC(=O)N1 89256,c1(C(=O)NC(C2CCCN(C(=O)C=CS(C)=O)C2)C)cc(C(F)(F)F)ccc1Cl 89257,C1(NC(=O)Cc2ccccn2)CCC2CN(C(=O)CCCCC(F)(F)F)CC2C1 89258,c1(C(=O)NC2(CC=C)CN(C(C3(OC)CCOCC3)=O)C2)cnc(S(C)(=O)=O)s1 89259,c1(OC)n[nH]c(NC(C2CN(C(c3cc(C)ccn3)=O)CCO2)=O)c1C#N 89260,N1(C(CSCC#C)=O)CC2(C(N3CCOC(CCF)C3)=O)CCC1CC2 89261,N1(C(c2cncc(C#C)c2)=O)CCC2CN(C(c3cccc(OC)n3)=O)CC12 89262,C1(n2cc(COCP(C)(C)=O)nn2)CCCN(C(=O)CN2CSCCSC2)C1 89263,N1(C(c2cn(C3(C)CC3)nn2)=O)CC(NC(=O)COC2CCOCC2)CC(O)C1 89264,CC1C(NC(C2CC(O)C2)=O)CC2CCC1N2C(C1(CO)CCC1)=O 89265,Cc1c(N(CC(C)(C)C(F)(F)F)C)nc(Cl)nc1O 89266,N1(C(C2(CC)CNC(=O)C2)=O)CC=C(C(=O)N(C)CC2(N(C)C)CCC2)C1 89267,C1(NC(c2ccc(COC)o2)=O)CCCCC1NC(C1CCCC1C(F)(F)F)=O 89268,C(CC(C(C)(C)C)NC(c1cc(F)cs1)=O)N(C(c1c(CC)n(C)nc1)=O)C 89269,C1(CNC(Cc2cccc(OC)n2)=O)CCC2(CCC2)C1NC(=O)C1CC1 89270,N1(C(CC(C)OC)=O)CC2CC(C1)CN(C(=O)CC1CCN(C)C1=O)C2 89271,C1(CC)CCC(F)(C(=O)OC2CN2Cc2ccc(F)cc2)CC1.OC.OC 89272,c1(COC(C)C)cc(C(=O)NCCN(C)C(C2COC(C)(C)CO2)=O)ccc1F 89273,C1(NC(C(CC)O)=O)C=CCCC1C(=O)NCCC1CCCC12CC2 89274,c1(C(=O)NC23C(CCN(C(C4(CC)CC4)=O)CC2)C3)cc(O)nc2c1CCCC2 89275,CC(O)CC(=O)NCC1(C(=O)NCCCC2CCCC2O)CC1 89276,C1(N(C(C(C)C2CCCC2)=O)C)C2CN(C(=O)CCc3ccc(N)cn3)CC12 89277,Cc1cc(F)c(C(=O)NC2CC(C)(NC(c3ccnc4c3CCC4)=O)C2)cc1F 89278,C1(C(=O)NCC(=O)NC)CCN(C(=O)CCN2CCOCC2)C1 89279,c1(C(N(C(CCNC(c2nc(C)oc2)=O)C)C)=O)cnc2n1CCC(C)C2 89280,N1(C(C2C(SC)CCC2)=O)CCC(C2(O)CN(C(c3coc(CO)c3)=O)C2)CC1 89281,c1(C(=O)NCC2CC(NC(C(C(C)O)N(C)C)=O)C2)ccc(C2CC2)c(F)c1 89282,c1(C(N2CCC(NC(C3(OC)CC3)=O)C(C(C)C)C2)=O)ccnc2c1ncn2C 89283,Cc1c(C(=O)NC2(C)CN(C(C3CCCN3C)=O)C2)cccc1Br 89284,c1(C(=O)NCC=CCNC(CC=CC=C)=O)cccc2nc(CC(C)C)[nH]c12 89285,Cc1c[nH]cc(C(=O)NC(C(C)NC(c2cn(C)nc2C(F)F)=O)C(C)C)c1=O 89286,c1(C(N2C3CC(NC(c4c(C)nncc4)=O)C3CC2)=O)cccc2c1ncn2C 89287,N1(C(CC(=O)OC)=O)CCC(CC(N)=O)(NC(=O)Cc2ccsn2)CC1 89288,C(=O)(C1CCc2cccc(F)c21)NCC(C1CC1)NC(c1c(C)noc1C)=O 89289,CCC(CCCC(=O)N(CC(O)(CC)CC)C)NC(=O)CC1CCCC(=O)C1 89290,N1(C(c2c(C)n(C)nc2)=O)CCC(C(N2CC(O)C(C)(C)C2)=O)C(C)(C)C1 89291,N1(C(c2n(CC)nc(C)c2)=O)CCC2CCC(NC(=O)C=CC3CCCN3C)C12 89292,N1(C(CCSCCC)=O)CCCC(C2CCN(C(=O)CC(F)F)CC2)C1 89293,N1(C(CN(C(C)=O)C)=O)CCC(C)(CC(=O)N(C)OC2CCCC2)C1 89294,N(C1CCCc2ccoc21)C(C1(NC(C(C)C2CCCO2)=O)CCC1)=O 89295,Cc1ccc(NCC(N2CC(CNC(=O)CN3CCCS3(=O)=O)CC2C)=O)cc1 89296,c1(C(N2CCC(NC(C=CCC)=O)(CO)C2)=O)nc2ncccn2n1 89297,C1(C)(CNC(C(c2cn(CC)nc2)=O)=O)CCCN1C(=O)CCOCC(F)(F)F 89298,C1(CNC(C2(C)CC2)=O)C=CC(NC(c2coc(Br)c2)=O)C1 89299,N1(C(C2CCC(C)N2C(=O)C(N2CCOC2=O)C)=O)CCc2cnccc2C1 89300,C1(C(=O)NC(C(C)NC(C=Cc2ccc(CC)cc2)=O)C)CCn2nnnc2C1 89301,N1(C(C(CC=C)c2ccccc2)=O)CCCCC2C1CCCN2C(=O)CSCC 89302,N1(C(=O)CCSC(F)(F)F)CCC(N(C(=O)CC2(CO)CC2)CCO)CC1 89303,c1(CCN2CCC(N)C2)ccc(OC(F)F)cc1F.CC(CCO)c1cn[nH]c1 89304,N1(C(c2c(C)c(F)cnc2)=O)CC2CC(C(=O)NCCCN=[N+]=[N-])C(C2)C1 89305,c12cc(ccn1)NC2=O.N1(CCN(CCC(=O)O)C)CCCCCC1 89306,c1(C(N2CCC(C(=O)NCC(C(CC)C)(C)O)C(C)C2)=O)c[nH]c2nccc-2c1 89307,C(=O)(CCC(C(C)C)NC(C1(C)CC(=O)C1)=O)Nc1ccc(C#C)nc1 89308,C1(CNC(CC2CCC(OCCC)CC2)=O)CCN(C(=O)C(C)SCC)C12CC2 89309,C1(CC(=O)NCC2N(C(CCCN(C(=O)OCC)C)=O)CC2)CCCC1(F)F 89310,N1(C(c2[nH]n(C)c(=O)n2)=O)CCC(F)C(NC(=O)CCN2CCCC2)C1 89311,c1(C(C(F)F)NC(=O)NC(C2CCOC2=O)C)cccc(Cl)n1 89312,N1(C(C2(C)CC=C(C)CC2)=O)CCN(C(C2(C#N)CCCOC2)=O)CC(O)C1 89313,c1(C(N(C2CCCC(NC(C3CC(=C)C3)=O)C2)C)=O)cnn2cc(C)cnc12 89314,O=CN1CCCC1C(N1CC2C(CNC(c3csnc3Cl)=O)C2C1)=O 89315,Cc1c(Cl)sc(Cl)c1C(N1CC2CC(NC(=O)CCc3ncc[nH]3)C1C2)=O 89316,C1(NC(C(C)CC2CC2)=O)CC2CCC1CN(C(c1ccc(=O)n(C)c1)=O)C2 89317,CCCCCCC(C)C(=O)NCC(CNC(=O)CCSCCCC)OC 89318,N1(CC(=O)N(CCCNC(C(C)N2CCCC2)=O)CCO)CCC(C)(C)C1 89319,CC1CCCn2c(C(N3CCCC(N4CC(O)C4)C3)=O)cnc21 89320,C1(NC(c2n(C)ccc2)=O)CCCCC1NC(c1ccncc1F)=O 89321,N1(C(C2C(CC)CCC2)=O)CC2CCCC(C1)N2C(c1ccc2cnsc2c1)=O 89322,C12(C(=O)NC3CCCN(C(c4ccc(NC)c(F)c4)=O)C3)CCCCN1CCC2 89323,N1(C(C(Cc2ccccc2)NC(=O)CN2CCCCC2)=O)CC(O)CC(F)(F)C1 89324,C1(C(N2CC(C)C(NC(=O)CC(=O)NC3CC3)C2)=O)C2CCCCCCC12 89325,c1(C(C)OC)nc(NC2(CO)CCCN(C(=O)C(C)C(C)COC)C2)cc(Cl)n1 89326,N1(C(=O)CCn2cncn2)CC2CCC(C1CO)N2C(=O)CC1CCCCCC1 89327,CC1CCN(C(C2CN(C)CCN2C)=O)CCN1C(C1CCCN1C=O)=O 89328,c1(C(C(=O)NC2CCCCN(C(CC(=O)NCC)=O)C2)C)cc2ccccc2o1 89329,CC1CN(C(=O)NCc2ccn(C(F)(F)F)n2)CC(C)S1 89330,C1(NC(c2ncn(C)c2)=O)CN(C(C2CC(=C(F)F)C2)=O)CC2(CCC2)C1 89331,c1(CC(=O)NCC2C3CN(C(C(C=C)(F)F)=O)CC32)noc2ccc(F)cc12 89332,N1(CC2CCc3nc[nH]c3CC2)CCCC1C1CCCN1CC 89333,C1(C(C(=O)OCC)C#N)CCCN(C(=O)Nc2cc(N)cnn2)C1 89334,Cn1cnc2cc(C(=O)NC3CC4(NC(=O)CC5(CO)CC5)COC3C4)ccc12 89335,C1(NC(Cn2cc(CC3(C)CCCC3)nn2)=O)COC2(CNC(=O)O2)C1 89336,C(C#Cc1ccccc1)N1CC(C)C(NC(=O)CCCC(N)=O)C1 89337,C(=O)(C1=NNC(=O)CC1)N1CCN(C(C=Cc2cc(OC)ns2)=O)C2C1C2 89338,C1(C(N2CCC(CNC(c3onc(COC)n3)=O)C2)=O)CCCCNC1=O 89339,O=C(CC(C(F)F)NC(=O)CN1CCCC1)NC1CC2OC1C1CC21 89340,c1(C(=O)NC2CC(N(C(CC(C=C)C)=O)C)C2)cnc(O)n(C2CC2)c1=O 89341,C1(NC(C=COCC)=O)CN(C(=O)Cc2ccc(O)cc2)CC1N=[N+]=[N-] 89342,C1(C(=O)NCC2(CNC(C(C(C)C)C)=O)CC2(F)F)CC(F)(F)C1(C)C 89343,c1(C(N(CC(C)(C)NC(c2nccc(C)c2O)=O)C)=O)cc2cccc(F)c2o1 89344,C#CCC(O)C(=O)NC(C)(C)CNC(=O)C(=Cc1ccccc1)NC(C)=O 89345,C12(NC(c3ncccc3F)=O)CCC(CC1)N(C(C1(F)C3CCCC13)=O)C2 89346,c1(C(N(C)CC2COCCN2C(C2SCCCS2)=O)=O)cccc2nc[nH]c12 89347,CC(C(=O)NCCCN(C(=O)Cc1ccc(Br)s1)C)C(F)(F)F 89348,c1(CNC(c2[n+]([O-])ccc(OC)c2)=O)ccc2c(c1)CN(C(=O)C(C)C(C)O)C2 89349,C1(CC(=O)NC2C(C)N(C(=O)Cc3csc(=N)[nH]3)CCC2)SC2=NCCN2C1=O 89350,Cc1c(C(N2CCC(N3CC(F)(F)C3)CC2)=O)cc([N+](=O)[O-])cc1[N+](=O)[O-] 89351,C1(CNC(CNC(C)=O)=O)CN(C(C2CC2C)=O)CC12CC2 89352,c1(C(=O)NC2CCN(C(C(COC)(F)F)=O)C2)ccc2c(c1)nc(C(F)F)n2C 89353,c1(OCC(=O)NC2CC2NC(c2ccnn2C2CCC2)=O)cccnc1 89354,N1(C(CCN(CCC)C(C)=O)=O)CCC(O)(CC)C1 89355,N1(C(c2cc(C3CC3)[nH]n2)C(=O)NCCOCC)CCC(C(C)(C)CO)CC1 89356,C1(CNC(C(c2n(C)ncc2)(C)C)=O)CN(C(C2CCC(C)CC2)=O)CCO1 89357,n1(CC)cc(C(=O)N(CCCCCCNC(=O)OC(C)(C)C)C)c(OC)n1 89358,n1(CC(=O)NC(CC)CN(C)C(c2cnn(C)c2OC)=O)cc(C)ccc1=O 89359,C1(NC(C(C)(C)OC)=O)(COC)CCN(C(=O)C(c2cccc(Cl)c2)C)C1 89360,C1(C(=O)NC(C2CC(NC(C=C(C)C)=O)C2)C)C2CCCC12 89361,c1(C(=O)NC2(CCNC(C3CCOC3)=O)CCCC2)cnc(-n2cccn2)cn1 89362,C1(CC(N2CCOC(CCNC(=O)CN3CCC3C)C2)=O)(OC)CCCCC1 89363,c1(C(C(=O)OC)OC(c2sccc2OC(C)C(=O)O)=O)ccc(Cl)c(Cl)c1 89364,C(CCC(C)NC(c1ccnn1CC1CCC1)=O)NC(C=C(CC)C)=O 89365,C1(C(=O)OC2CCC(C)CC2)(N(C)C)CC2(CC(F)C2)C1 89366,c1(C(=O)NC(C)CCNC(c2nnn(C)c2C(F)F)=O)cc2n(c1)CCC2 89367,C1(N(CC)Cc2cccs2)CCN(C(c2cnn(C)c2)C(=O)NCCCF)CC1 89368,C12(C3CC3)CN(C1)C(=O)N2.C1(c2ccccc2)(COC)CCOC1 89369,C#Cc1cnn(C)c1C(N1CCOC(C(=O)NC(c2cn(C)nc2C)C)C1)=O 89370,C1(NC(C2(NC(=O)CC34CCC(CC3)C4)CSC2)=O)COCC1C1CC1 89371,c1(N2CCCC(C)(N(C)C)C2)nc(NCC2(CCO)CCOC2)c2ncsc2n1 89372,c1(C(=O)NCCC(CNC(c2ccc(C)cc2Cl)=O)(C)C)ccn2nncc2c1 89373,c1(C(=O)NCC(CC=C)NC(=O)C(C)(CC)CCC)ccc(CC)c([N+](=O)[O-])c1 89374,c1(CC(N2CC(C(C)NC(c3cccc(OC)n3)=O)C2)=O)ccc(C)c(F)c1F 89375,c1(COC)nn[nH]c1C(=O)NCCNC(=O)C(c1ccncc1)c1ccccc1 89376,C12(C(=O)OCC)COC(C(=O)NCCC3CN(C(=O)C(C(C)C)N(C)C)C3)(C1)C2 89377,c1(-c2c(C)ccs2)csc(=Nc2cccc(C(N)=O)c2)n1Cc1ncoc1C(C)C 89378,C(=O)(C(C(C)O)NC(=O)CCCCN(C)C)NCCOCCC=C 89379,c1(C(C)=O)cc(C(=O)N(CC(C)CNC(=O)Cc2cnc(C)o2)C)co1 89380,CC1CCC(C)(C(N2CCC(=CCNC(=O)CC3(C)OCCO3)CC2)=O)C1 89381,C1(C(=O)NC(CC)CN(C)C)CN(C(c2sccc2OC)=O)C(C)(C)C1 89382,Cc1cc([N+](=O)[O-])ccc1C(=O)Nc1nnn(C(C)(C)C)c1C(N)=O 89383,C1(OC)CC(N=c2[nH]c(=NC(C)c3ccncc3F)c3ncccc3[nH]2)C1 89384,N1(C(CNC(c2ccoc2)=O)=O)CCN(C(c2cc(O)ncn2)=O)C2COCC12 89385,n1(C(C)C)cc(Br)c(C(=O)NCC(O)CNC(=O)CSc2ccncc2)n1 89386,c1(CC(=O)NCC2CCC2NC(C2COC2)=O)ccc2c(c1)OCCCO2 89387,Cc1cc(C(=O)NCC(O)CNC(=O)C=Cc2cnc(C)s2)n(C2CC2)n1 89388,CC(C(=O)NCc1nc(C(=O)NC2(CC3CC3)CC2)co1)C(F)(F)F 89389,C1(C(=O)NCCNC(=O)NCC)CN(C(C2C=CCS2)=O)CC1(C)C 89390,C1(C)(C(N2CC(C(C)OC)C2)=O)CCN(C(=O)C=C(C)C(C)C)C1 89391,N1(C(c2c(CC)c[nH]c2)=O)CCC2CCN(C(c3cc(C)on3)=O)C2C1 89392,N1(CC)CC(C(=O)NC2CCC(NC(c3nc(O)sc3C)=O)CC2)CCC1=O 89393,c1(C(=O)NCc2cn(C)nc2C(F)F)c(F)ccc(O)c1F 89394,c1(CCNC(=O)NC2CN(CCN(C)C)C(=O)C2)ccc2occc2c1 89395,CC1(C)CCCC(C)(C)C1C(N1CCCC1CNC(C1CCN1C1CCCC1)=O)=O 89396,C12(CNC(C(C(C)C)F)=O)CN(C(C3CC4(CCC4)CO3)=O)CC(F)(C1)C2 89397,c1(C(N2C(C(N(CCCCO)CC)=O)CCC2)=O)ccc(C)cc1Cl 89398,C12CCC(CC1)C(=O)N2CC.C(=O)(C(C)Cc1cccnc1)NC1CC(CF)C1 89399,C(=O)(C(CCOC)OC)NCC(C)N(CCOC)C(c1nc(C(=O)OC)oc1C)=O 89400,CC(C)C(CCC(=O)NCC(C)CN(C)C)NC(c1ccc(O)nc1)=O 89401,N1(C(C(C)OCC#C)=O)CCOC(CC(=O)NCCc2ocnc2CO)C1 89402,c1(NC(C23C(CN(C(c4n(C)ccc4)=O)C2)C3)=O)c(C)ccc(C(=O)O)c1F 89403,c1(C(=O)NCC(c2ccccc2)CNC(C=NOC)=O)c(N)cc(Cl)cc1F 89404,c1(CN(C(CC(=O)OCC)C)C)cc(C)c(C)cc1O 89405,C1(NC(C23CCC(NC(C(COC)N(C)C)=O)(CC2)C3)=O)CC2(C1)CC(C#N)C2 89406,C1(CCNC(=O)CC2CCNC2=O)CN(C(C2(O)CCCCC2)=O)CCO1 89407,N1(Cc2c(C)n[nH]c2C)CCCC2(CCCN(C(c3ncsc3C)=O)C2)C1 89408,Cc1cccc(Br)c1C(N1CC(NC(=O)C(C)Cc2ccccn2)C(O)C1)=O 89409,N1(C(C2CCC(=C)CC2)=O)CCCC1C1CCCCN1C(=O)Cc1cnoc1 89410,CC1CC(C(N2CC(NC(c3nc[nH]c3C(C)(C)C)=O)C2)=O)C1(C)C 89411,N1(C(CN2C(C)CCC2)=O)CC(N(C(=O)Cn2ccc(O)nc2=O)C)C(C)(C)C1 89412,c1(C(=O)NC2CCCC2C(F)F)c(Cl)ccc2ccncc12 89413,N1(C(CC2CC(C)C2)=O)CCNC(=O)c2c(Br)cccc21 89414,Cc1c[nH]nc1CNC(=O)CC1CCC(NC(=O)C(C2CCOCC2)O)C1 89415,C(=O)(C(C)C(O)C(C)C)N1CC(CCNC(c2c(C)ncnc2C)=O)(OC)C1 89416,CC(CO)C(C)N=c1ccnc(NCc2cccc(Cl)c2Br)[nH]1 89417,N1(C(c2c(C)scn2)=O)CCCC(C(N2CCCC2CNC(N)=O)=O)(CO)C1 89418,N1(C(C2=NOC(C)C2)=O)CCCN(C(=O)C(C)Cc2ccncc2)C(C)C1 89419,CC(C)(O)C(CCO)NC(C1CC2(CC2)CN1C(=O)CCc1cncs1)=O 89420,N1(C(C(C(C)C)C(C)NC(=O)C(O)CC(N)=O)=O)CCC(O)(C2CC2)CC1 89421,[N-]=[N+]=NC1CCN(C(C2CN(C(=O)COCC(F)F)CC23CC3)=O)C1 89422,N(C(=NCC1CCC(=O)NC1)N1CCC(CCC#N)CC1)C(COC)C 89423,C1(C)(NCCCn2c(C)ncc2)CC(C#N)C1 89424,c1(CC(C(=O)NCCC(C)NC(c2cn(CC)nc2)=O)O)cc(Cl)cc(Cl)c1 89425,C1(CNC(CC2N(C)CCC2)=O)CC2(CCC2)CN1C(=O)C(c1ccccc1)=O 89426,N1(C(C(CC#CC)NC(c2ccncc2O)=O)=O)CCC2(C1)CN(C)C2 89427,C(=O)(C1=CCCOCC1)NCC1(F)CCN(C(c2cc(N)cc(F)c2)=O)C1 89428,N1(C(c2nc(C(C)=O)sc2)=O)CC(NC(C2CCC(C)(C)O2)=O)C2(CC2)C1 89429,N1(C(c2n(CC)ncn2)C(=O)NC2CC2)CC(SC)CC12CCOCC2 89430,c1(CC)ncc(C(N2CCCC(N(C(c3snnc3C)=O)CC)C2)=O)c(C)n1 89431,Cc1nc(C(=O)N(C)CC2CCCN2C(=O)C(C2CCCO2)C2CC2)c(C)o1 89432,c1(C(=O)OC(COC)C(C)C)cc(O)nc(COC)n1 89433,C=CC1(CC(=O)OCC(=O)NC2CC2C#N)CCCCC1 89434,S(=O)(=O)(c1cccc2c1OCCC2)N1CC(O)CC(OC(C)(C)C)C1 89435,N1(C(C(CN(C(=O)C=CCF)C)(C)C)=O)CCC2OCCCC2C1 89436,c1(C(N2C(C)CCC(NC(CCOC)=O)C2)=O)cc2c(OC)[nH]c(=N)nc2s1 89437,C(CCCCC(=O)NC1CC=CCC1C(=O)N(CCC)C(C)C)=CC 89438,c1(C(=O)NC2(C)CN(C(C(C)(C3CC3)SC)=O)C2)ccc(=O)n(-c2ccccc2)c1 89439,N1(C(c2ccc(SC)cc2)=O)CCC2(C)CN(C(=O)CCOC(C)=O)CC12 89440,Cc1ccc(NC(C2(C(C)NC(=O)OC(C)(C)C)CC2)=O)cc1N=[N+]=[N-] 89441,N1(C(c2c(SCC=C)cccc2)=O)CC2(C1)CN(C(C1CCC3CC3C1)=O)C2 89442,N1(C(CCC=C)=O)CCN(C(=O)Cn2cc(Br)ccc2=O)CC1CC1CC1 89443,C1(C(N2C(CC=C)CCCC2)=O)CN(C(C2CCCN2C)=O)C(C)(C)C1 89444,CCC(CNC(C1CCCCN1C(=O)C(n1ccnc1C)C)=O)C(C)C 89445,C=CCC(CNC(=O)C=NOC)NC(C1CCCN1C(=O)Cc1ccccc1)=O 89446,c1(C(N2CCC(CNC(=O)CC(O)C3CCCC3)C2)=O)cc([N+](=O)[O-])cnc1O 89447,N1(C(C(n2cc(CCN(C)C)nn2)C)=O)CC2CC2(CO)C1 89448,C1(OCC)CN(C)C(C)(C(N2CCC(CN(C)CCc3ccccc3)CC2)=O)C1 89449,C=C(CN=c1[nH]cnc(NCc2cc(CC)on2)c1C)C(C)(C)C 89450,CCC1=C(C(=O)NCC2CN(C(C3CCCN3C(C)=O)=O)CCN2C)CCCO1 89451,N1(C(C(C)CF)=O)CCC2(CC1)CCN(C(c1cc(F)ccc1O)=O)CC2 89452,c1(CCC(=O)N2CCOC2)nc(O)n[nH]1.c12ccc(s1)Cc1cn(nn1)NC(=O)CSC2 89453,c1(C(N(CCC2CCN(C(C3(C)CC(=C)C3)=O)CC2)C)=O)ccc(C)c(C)c1Cl 89454,Cc1cc(C(=O)NCCCCN(C(=O)Cc2ccnn2C)C)c2cnn(C)c2n1 89455,N1(C(c2c(OC)nccc2)=O)C2CCC(C2)C1C(=O)Nc1nc(Br)cnc1Cl 89456,n1(CC(=O)NCC2CCN2C(=O)CNC(=O)NC2CC2)cc([N+](=O)[O-])cn1 89457,N1(C(C(=O)NCC)=O)CCC2OCCN(C(=O)CCOCc3ccccc3)C2C1 89458,N1(C(C(CO)NC(N)=O)=O)CC2CC1CN2C(c1cc(Cl)ccc1Cl)=O 89459,CCC(C)CC(=O)C(=O)NC(CO)C(=O)NCC1CCc2nccn21 89460,C(=O)(CC(C)n1ccnc1)N1CC(N(C(CC)CC)C(=O)CNC(N)=O)C1 89461,C1(OC)CC2(C1)CC(C(=O)NCCN(C)C(c1cncc(F)c1C(F)(F)F)=O)C2 89462,C#Cc1ccc(CNC(=O)C(O)CCNC(=O)CC2CC(C)C2)cc1 89463,C(CCCCC(=O)N1CC(NC(=O)CC2CC2(Cl)Cl)CC1(C)C)OCC 89464,C#CCCC(C(=O)N1CCC(N=[N+]=[N-])C1)NC(=O)CC1CC(SC)C1 89465,Cc1nc(NCCN(C)C(C)C)cc(=NCCC(C)C(C)C)[nH]1 89466,C(C(C)(C)C(=O)N1CC(F)CC1C(N1CC(S(C)=O)C1)=O)N(C)C 89467,C1(NC(CC=C)=O)CN(C(c2ccc(C(N)=O)o2)=O)CC1CO 89468,C1(NC(c2cn(CC)nc2)=O)(CO)CCN(C(=O)C(O)COC)C1 89469,N1(C(Cc2ncn(C)c2)=O)CC2CC1(CNC(C1CC13CCOC3)=O)C2 89470,c1(C(N(CC(C)NC(C(C=C)CC)=O)C)=O)ccn(C)c(=O)c1 89471,C1(O)(CN(CC#C)C(c2cccc(-c3ccccc3)c2)=O)CCN(C(=O)CO)CC1 89472,N1(C(CC(C)C)=O)CC2CC1CN2C(C1OCCN(C)C1=O)=O 89473,CC1(C)C(CNC(C2(c3cc[nH]n3)CC2)=O)CCN1C(C1CCNC1=O)=O 89474,c1(CNC(=O)NCCSCC(F)F)ccc2c(c1)CCO2 89475,N1(C(c2cc(C)[nH]n2)C(=O)NC(CC)(C)C)CCC2CC(CN(C)C)CCC2C1 89476,c1(C(=O)NC(CC=C)CNC(=O)C(c2ccccc2Cl)O)cnc(CC)nc1C 89477,C1(NC(C2N(C(C)C)CCC2)=O)CCC2CN(C(c3cnnc(O)c3)=O)CC2C1 89478,C(C1c2ccsc2CCN1C(C1(C2CC2)CC1)=O)NC(Cc1nc(CC)sc1)=O 89479,Cc1cn(CC(=O)NC2CC23CCC(NC(=O)C(C)O)CC3)c2ccccc12 89480,C(C)(CO)(C(F)(F)F)NC(c1cn(CCNC(c2cc(OC)n(C)n2)=O)nc1)=O 89481,C1(OC(C)C)CCN(C(c2cc(CNC(=O)C=CC(F)(F)F)cs2)=O)C1 89482,C1(NC(CN(CC)CC)=O)CC2(CCCCN2C(c2ncccc2CSC)=O)C1 89483,c1(C(CC)C)nccc(=NCC23CC(NC(c4[nH]ccc4COC)=O)(CO2)C3)[nH]1 89484,C1(C(C(=O)O)Nc2ccc(C(=O)OC)cc2)CC(=O)N(C)C1c1cnn(C)c1C 89485,C(=O)(C1=CC2(CCOCC2)C1)NC1CC(C)N(C(c2cc(C(N)=O)cn2C)=O)C1 89486,N1(C(C(F)=C(C)C)=O)CCOC(CCNC(=O)CCc2nccn2C)C1 89487,C12(C(N(CCC#C)C)=O)C(NC(c3ncncc3C)=O)C3CC1C2C3 89488,N1(C(C(CC)CCOC)=O)CC2CCOC2(CNC(=O)Cc2sc(C)nc2C)C1 89489,Cc1c(C(N2CC(CO)OC(CO)C2)=O)[nH]c2cc(Cl)ccc12 89490,CCS(=O)(=O)c1ccc(Cl)c(C(=O)NCC2CCN(C(c3cc(F)c[nH]3)=O)C2)c1 89491,C1(C(N2CC3C(NC(C4(OC)CC4)=O)(C3)C2)=O)CCCCC12OCCO2 89492,N1(C(COCP(C)(C)=O)=O)CCC2CCN(C(C3(CN(C)C)CC3)=O)C2C1 89493,c1(CNC2CCC(C(=O)NCC(C)O)C2)c(Cl)cc(F)cc1Cl 89494,Cc1cc(C(=O)N(CCCN(C)C(C2CCOC2)=O)C)c2c(n1)CCCC2=O 89495,N1(C(C(C)NC(C)=O)=O)CCN(C(=O)CCCc2nccs2)C(c2cn[nH]c2)C1 89496,N1(C(c2cccc(NC)n2)=O)CCC2(CCCCC2NC(=O)CC(C)C2CC2)C1 89497,S(=O)(=O)(c1ccc(NCc2cnccn2)c(Br)c1)N1C(C)C(C)(C)CC1 89498,C12(C(=O)NC(c3ccccc3)CNC(Cc3cc(C)no3)=O)CC3CC1C2C3 89499,c1(C(CCO)NC(c2n(CC)nnn2)(C)COC(C)C)ccc(F)cc1.C1CO1 89500,C1(CNC(C(C)=C2CCC2)=O)CN(C(c2cccc(Br)c2)=O)CCC1(C)C 89501,Cc1c(C(=O)NCC2CCCN(C(=O)C=CC3CCCC3)C2)nn(C)c1C1CC1 89502,c1(C(N2CCN(C(C3CC4CCCCCC34)=O)CC2)=O)cc(O)ccc1Cl 89503,C(C(C)(C)C(=O)NCCF)N(C(=O)C(C1CCOCC1)=O)C 89504,c1(C(=O)NCC2CC2NC(C2(Cl)CCC2)=O)ccc2c(n1)CCC2 89505,c1(C(N(CC(CC)NC(=O)C(CC)N(C)C)C)=O)cc(C)c2c(O)n[nH]c2n1 89506,C(CC1=CCCCCC1)NCC1(CO)CCN(Cc2ccc(F)cc2)C1 89507,c1(C(C)C)cc(=NC2CC(NC(=O)CCNC(=O)C=CCl)C2)[nH]c(C(C)C)n1 89508,N1(C(C(CC=C)(C)O)=O)CC(C(N2CCC(C)(CCO)C2)=O)C2(CCC2)C1 89509,C(=O)(CC1=CCCC1)NC(C1CCN(C(c2conc2C(C)C)=O)CC1)C(C)C 89510,CC1(C)CCC=C1C(=O)N1CCCN(C(=O)Cc2ccc(F)c(Cl)c2)CC1 89511,c1(C(=O)NCCN(C(C(=O)NC(CC)C)C)C2CC2)ccc2cccc(F)c2n1 89512,N1(C(C(N2CCCC(O)C2)C)=O)CCCC(C2CC2NC(=O)Cn2cnnn2)C1 89513,c1(C(N(C2CCN(C(=O)CCc3cccnc3)C2)CC)=O)ccn(C(C)(C)C)c1 89514,c1(C(=O)NCc2cccc(C(=O)NC(CC(=O)OC)C)n2)c(O)cccc1F 89515,N1(C(CC(CNC(=O)C(=CC2CCCC2)C)OC)=O)CC2CC1CC2CF 89516,c1(C(=O)NC(CCNC(c2ccc(CC)[nH]2)=O)C)ccc2c(=O)n(C)cnc2c1 89517,Cn1ncc(C(N2CC(CNC(=O)CCOCC(F)(F)F)C(O)C2)=O)c1Cl 89518,c1(C(N2CC(CC(C)NC(COC(CC)C)=O)C2)=O)cc(=O)c(O)c[nH]1 89519,C(CCNC(C1(NC(C2C(C)(C)C2(C)C)=O)CC(O)C1)=O)(C(C)C)OC 89520,C(CC(=O)N(C)CC1COCCO1)(C(F)(F)F)NC(C1C(C(C)C)C1)=O 89521,C1(C(CNC(C2(CC)CCC2)=O)C)CCN(C(c2c(C)nsc2C)=O)CC1 89522,Cc1ccnc(CN2CCCC2CCNC(c2cccc(-c3nn[nH]n3)c2)=O)c1 89523,c1(NC2(C3CN(C(C4C5CCCC45)=O)C3)CC2)ccc2cnccc2c1[N+](=O)[O-] 89524,Cc1nnc2cnc(C(N3CC4CC3CCC4NC(=O)CC(C)(C)O)=O)cn12 89525,N1(C(C(C)Cc2cnn(C)c2)=O)CC2(CCCCN2C(C2CCC(CN)C2)=O)C1 89526,c1(C(N2CCC(N(C(=O)CC(F)F)C)C2)=O)ccc2c(c1)ncn2C 89527,N1(C(=O)Nc2c(Cl)cnc(SC)n2)CCCC2NC(=O)CCCC12 89528,C1(C)(CNC(C=CCCC)=O)CCCN(C(=O)C=Cc2nc(C)cs2)C1 89529,C(=O)(C(CC)C(C)(C)CC)NC(CC(=O)NC(CCCC)C)(C)C 89530,c1(CC)c(C(=O)NCCCCNC(=O)C(O)(CC)c2ccccc2)nnn1C 89531,c1(NC(=O)CCC2CCCO2)csc(CC(=O)Nc2ccco2)n1 89532,Cc1ccccc1NC(=O)C(N1CCOC(C(=O)N(C)C)C1)c1ccc(Cl)s1 89533,c1(-n2cc(CCC#N)nn2)ccccc1CC(N1CC(C(=O)O)C2CC12)=O 89534,c1(N(C(N(C)C)=O)C)ccc(C(=O)N(C2CC2)Cc2cn(CCCCO)nn2)cc1 89535,Cc1cc(C=CC(=O)NC(C)C(C)NC(=O)C(C)(Cl)Cl)ccc1C(F)(F)F 89536,C1(CCC)(NC(c2coc(C(C)C)n2)=O)CCCN(C(c2cncc(N)c2)=O)C1 89537,c1(C(=O)NC(C(=O)O)C2CCOC2)cccc(S(=O)(=O)NCCCO)c1 89538,N1(C(CCOC(C)=O)=O)CCC(F)(CNC(c2ccn(CC(F)F)n2)=O)C1 89539,CC(C)CC(CNC(=O)C=Cc1cncn1C)NC(C1CN(C)CCO1)=O 89540,c1(OC)ccc(C(=O)N(CC(C)CNC(=O)C=Cc2cncs2)C)cc1OC 89541,C=CCC(C(=O)N1CC(O)CC1C(=O)NC1(C2CCCO2)CC1)OC 89542,CC1C(C=CC(N2CC(O)(CNC(c3ccc(C(N)=O)o3)=O)C2)=O)C1(Cl)Cl 89543,C1CCNC(=O)C2(CC2)CCN1CCC.C(C)(C)(C)O.C(N)=O 89544,c1(C(=O)NCC23N(C(C(CC)CC)=O)C(CC2)CC3)c(Cl)ccc2ccncc12 89545,CCC(CC)C(F)C(=O)NC(CCC(=O)N(C1CCC1C)C)C(C)C 89546,C1(CC(C)NCC2CC(CC(C)(C)C)C2)CCN(C(=O)CC(Cl)Cl)CC1 89547,CCC(C)(CNC(C1CC1F)=O)NC(c1cc(CF)on1)=O 89548,c1(OC)ccc(CC(=O)NC2CCCC(C(=O)NCc3nc(C)no3)C2)c(F)c1 89549,c1(C(=O)NCC2(NC(C3CC3c3ccsc3)=O)CCC2)cccc2c1CCCN2 89550,c1(OC)cc(F)c(-c2ncccc2C(=O)NC(c2cccnc2)C2CC2)c(F)c1 89551,C1(CNC(CC(C)(C)O)=O)C2CCCCCC12.C12CCCCC1NC2=O 89552,C1(C)(Nc2ccc(CNC(CCC(=O)OC)=O)cc2)CCCS1(=O)=O 89553,N1(C(CC(CC)NC(C=CCCC)=O)=O)CC(C)CCCC1C 89554,N1(C(C(COC)C)=O)CCC(C(=O)NCC2CC23CCOC3)CC1C 89555,N1(C(C2(CSC)CC2)=O)CC(CO)(NC(C2CC(=O)N2)=O)C1 89556,C=C1Cn2c(C(=O)NCC3(C(N)=O)CN(C(=O)Cn4cc(CO)nn4)C3)nnc2S1 89557,c1(NCc2cccc(C(N)=O)c2)ccc(Br)c2c1C(=O)NC2=O 89558,c1(C(C)C)occc1C(=O)NC1CN(C(C2CC2C(F)F)=O)C1.n12cnc(n1)C2 89559,c1(CC(=O)NCCC(C)NC(=O)C=Cc2cnccn2)cn2ccsc2n1 89560,CN1CCOCC2(COCCN2C(=O)NC2CCC3(COC(C)C3C)O2)C1 89561,C1(C(=O)Nc2cccc(CNC(C(CCC)OC)=O)c2)COc2ccccc2C1 89562,C1(NC(C(C)=C(CC)C)=O)CC(N=c2[nH]cnc3c(COC)nsc23)C1 89563,c1(CC)c(N2CCN(C3CCN(C(=O)C=CCF)CC3)CC2)nc(C)nc1Cl 89564,C1(C)(C(N2CC(OCCNC(C(c3cccnc3)OC)=O)C2)=O)C(C)(C)C1(C)C 89565,c1(C(=O)NCC2CC(c3ccccc3)CO2)ccc(Br)cc1 89566,N1(CCC(=O)NCCCN(C(c2cnc(C)o2)=O)C(C)C)CCCCC1=O 89567,C1(C(=O)NCC2CC2NC(=O)C(F)OC(F)(F)F)CCC2(CC1)CC(O)C2 89568,C1(C(=O)NC2C(F)CCN(C(CC(C=C)(C)O)=O)C2)CN(CP(C)(C)=O)C1 89569,C(CC(C)CCNC(C1CCN(C(N)=O)CC1)=O)NC(C(N1CCOCC1)C)=O 89570,c1(OC)c(-c2nc(NC(c3csnn3)=O)cs2)cccc1C 89571,C1(C(=O)NC(CC=C)CO)CC(N=[N+]=[N-])CN1C(=O)C(O)CN(C)C 89572,C(=O)(C(CCSC)NC=O)NCCCCCN(C(CC)=O)C 89573,CCC(CC)CC(F)C(=O)NC(CNC(C1(C)CCOC1)=O)CCOC 89574,CN1CCCC1C=CC(N1CCOC(CCNC(=O)CSc2n[nH]c(O)n2)C1)=O 89575,C1(C(=O)NC(CNC(CN(S(N(C)C)(=O)=O)C)=O)(C)C)CN2CC3CC2(CO1)C3 89576,c1(SCC2(C(N3CCC(NC(CC(C)SC)=O)C3)=O)CC2)ccc(Br)cc1 89577,N1(C(c2c(OC)scc2)=O)CC2CN(C(=O)CN(C3CCC3)C)CC2(C)C1 89578,c1(C(=O)NCC2N(C(CCOCC#C)=O)CC(C)CC2)cccc2nonc12 89579,N1(CCCC)CCN(C(=O)CC2CCCCN2C(=O)Cn2cccn2)CC1 89580,C1(NC(C=CC(=O)Nc2cccc(C)c2)=O)COCCN(C(C2CCC2C)=O)C1 89581,C1(NC(=S)Nc2ccncc2)CC2CCC(C1)N2N(c1ccc(F)cc1)C 89582,c1(C(C(=O)NCCCCCC)N(C)CC2CCOC2)cc(C)nc(C)n1 89583,C(CS(=O)(=O)C(C)C)NC(=O)NC(C)CC1(O)CCOCC1 89584,Cc1c(CNC(=NCCNC(=O)Cc2ccccc2)NC2CC2C)c(Cl)nn1C 89585,c1(N2C(C)C(NC(c3ccc(CO)cn3)=O)CCC2)ncc(C#N)cc1Cl 89586,C(C)(CC(=O)NC1C2CC1N(C(c1ccc(CO)s1)=O)C2)(C(F)F)N(C)C 89587,c1(CC)ccc2cc(C(=O)NCC(C)CNC(C3(c4cc[nH]n4)CC3)=O)[nH]c2c1 89588,CC1(C)CN(C(C2CCCN(C3CCCCC3)C2)=O)C1c1cccnc1 89589,C1(NC(c2cn(CC3CCOC3)nn2)=O)CC12CCN(C(c1cnns1)=O)CC2 89590,c1(CC)ccccc1C(CNC(C1CCC2CC12)=O)NC(C1(CCO)CC1)=O 89591,C#Cc1ccc(CC(=O)NCCN(C(=O)C(=Cc2cccnc2)C)CC(C)O)cc1 89592,C1(C(=O)NCC(C(C)C)NC(C2CCCCC2)=O)CCCCN1C 89593,CCCC(C)CCCC(=O)Nn1cc(CC2(Cc3cc[nH]c(=N)c3)CC2)nn1 89594,C1(CNC(c2ccon2)=O)Cc2ccccc2CN1C(=O)CCOC1CC1 89595,c1(C(N2CC(CC=C)(NC(=O)Cc3ccsn3)C2)=O)c(C)cccc1[N+](=O)[O-] 89596,N1(C(COCC(C)C)=O)CC(NC(=O)CCCn2ccccc2=O)CC2(CC2)C1 89597,N1(C(C(C2CCC2)OCC)=O)CCc2ccc(C(=O)NC(CC)CO)nc2C1 89598,c1(CNC(C(CC)(C)C#N)=O)ccc2c(c1)CN(C(=O)Cc1ccns1)C2 89599,N1(C(C(C(CC)C)NC(=O)C=Cc2cocn2)=O)CC(F)(F)C(F)(F)C1 89600,Nc1c(C(N2CC3CC(NC(=O)COc4ccc(F)cc4)C2C3)=O)cccc1F 89601,C1(NC(=O)C2=CCCCC2)CCCC12CN(C(c1ccn(CCO)c(=O)c1)=O)C2 89602,C(=O)(C#CC(C)(C)C(F)F)NC1C(NC(C#CC(OCC)OCC)=O)CC1 89603,c1(C(=O)NCC2N(C(Cc3nnc(C)o3)=O)CCN(C)C2)cccc2c1CCC2 89604,c1(C(=O)NC2CCN(C(c3c(OC)ccnc3)=O)CC2)cnc2cnccc2c1 89605,C1(C)(C(=O)OCC)CCN(C(C(=O)NC2CC2)C(C)C2CCCOC2)C1 89606,CC1(CNC(c2ncoc2Br)=O)CCCN1C(C1CC(F)C(=O)N1)=O 89607,C1(C(=O)N(C(C)C(=O)N(C(C)COC(C)=O)C)C)(CC)CCNC1=O 89608,c1(C(=O)OCC)cccc(NC(=O)Nc2cnc(OCC(C)C)cn2)c1 89609,c1cc(=NCCCc2nccs2)[nH]c(NC2CCC(C3CC3)C2)n1 89610,c1(C(=O)O)cccc(CN2CCC(F)(C(N3CC(F)C(F)C3)=O)CC2)c1F 89611,CN1CC(O)(CNC(C2CCC(CNC(c3cc(C(N)=O)[nH]n3)=O)O2)=O)C1 89612,CC1CCN(C(=O)C(C)(C)N2CCCC2)CCN1C(C1CC2(CCCCC2)C1)=O 89613,N1(C(C(CC)N(C)C)=O)CCCC(CN(C)C(c2csc(COC)n2)=O)C1 89614,c1(C(N(CCCNC(C(CCOC)C)=O)C)=O)cnc2nc(O)nc(O)c2c1 89615,c1(CC(=O)NC2C(OC)CN(C(c3ccsc3OC)=O)C2)cc(F)ccc1O 89616,C1(CNC(Cn2c(=O)sc(C)c2C)=O)CN(c2nncs2)CCC12CCOC2 89617,N1(C(C)CC2CCC(=O)N2)CCC(CCNC(C2CCS(=O)(=O)C2)=O)CC1 89618,c1(C(N(CC(CNC(C2(CC)CC2(F)F)=O)O)C)=O)nn(C)c2c(=O)[nH]cnc12 89619,c1(C(N2C(C)CCC(NC(c3c(C)cn(C)n3)=O)C2)=O)cnc2ncccc2c1 89620,c1(CNC(C(F)=C(C)C)=O)ncoc1C1CN(C(C2CC(C)CO2)=O)C1 89621,C1(CN(C(=O)CCC2CCCC(=O)N2)C)COCCN1C(C1CC2(CC2)C1)=O 89622,c1(CC)ccc(N)c(C(=O)NCCN(C(=O)COC(F)(F)F)CC)c1 89623,c1(C(C(=O)NC(C(=O)NCC2(CCNC(C)=O)CC2)=O)C)cccnc1 89624,Cc1nn(C)c(N2CCOCC2)c1CN1CCCN(c2ncc(C(=O)O)s2)CC1 89625,N1(C(CN2CCCC(CC)C2)=O)CC2(CCCC2NC(C2C=C2C)=O)C1 89626,N1(C(C2C(C)C2)=O)CCC(OCCCNC(C2CC2c2ccoc2)=O)CC1 89627,C(CC(C(=O)NOCC1CCCC1)OC)NC(c1c(CC)[nH]cc1)=O 89628,C1(C(=O)NC(c2ccnn2C)C(N2CC(OC(C)C)C2)=O)C=CC=CC=C1 89629,CCC(C)(C)OCC(=O)NC1CC1CNC(=O)C=C(C)C(F)F 89630,C(c1cc(Cl)ccc1Cl)=CC(=O)NCC1(NC(=O)Cn2nccn2)CCOCC1 89631,C1(O)(CN(C(C(C)C2CCOC2)=O)C)CN(C(c2cnn(CCO)c2)=O)C1 89632,N1(C(C2(OC)CCCOC2)=O)CC2CC(NC(=O)Cc3n[nH]c(C)n3)C(C2)C1 89633,Cc1ccc(CNC(C)CCc2ccc(Br)cc2)c(Br)c1 89634,C12(NC(C(C)=CC)=O)CCCC1CN(C(c1cnn(CCC)c1Cl)=O)C2 89635,N1(C(CC)=O)CCCC(C(=O)NC2CCCC2NC(c2ccnn2C(F)F)=O)C1 89636,N1(C(c2c(CNC(c3c(CC)noc3)=O)occ2)=O)CC2CCC2(OC)C1 89637,C1(C(=O)NC2C(NC(COc3cccc(CC)c3)=O)CCC2)C(F)(F)C12CCC2 89638,C1(CNC(c2n(C)ncc2)=O)CC(F)CN1C(c1ccnnc1)=O 89639,c1(C(N2CCC(NC(c3cc(-c4cccs4)[nH]n3)=O)C2)=O)cc(F)cc(F)c1 89640,C1(CNC(CCC=C)=O)CN(C(=O)C(C)CCO)CCC12CCOC2 89641,c1(NC(CNC(c2c(CC)cno2)=O)=O)cccc(C#N)c1 89642,O=C(CCCC1CCC1)NCCn1cc(C(N2CC(c3cc[nH]n3)C2)=O)nn1 89643,N1(C(c2ccc(CC)cc2)=O)CCC(NC(C2COCC2(C)C)=O)C(O)C1 89644,C1(C(N(C2CCN(C(c3csc(O)n3)=O)C2)C)=O)CCS1(=O)=O 89645,C1(C(=O)NCCCN(C(CCC(CC)OC)=O)CCO)CCCC(C)(C)CC1 89646,N1(C(CC)CO)CC(=O)N(CC(=C)F)C1 89647,c1(C(N2C(CCCNC(c3n(CC#C)cnn3)=O)CCC2)=O)cccc(CC)n1 89648,N1(C(C(F)OC)=O)CCOCC(CNC(c2cnoc2)=O)C1 89649,N1(C(CCn2cc(-c3ccc(C)cc3)nn2)=O)C(C)CC(c2ccccc2)C1C 89650,C(=O)(C(O)CC(C)C)NCC1(CNC(COC(CC)(C)C)=O)CC1 89651,Cc1cc(C(=O)NCC2CC(F)(CNC(=O)CC(C)F)C2)ns1 89652,C1(C)(C(=O)NCCCOC)CCCN(C(=O)Cn2nc(C)cc2C)C1 89653,C1(CNC(C(=Cc2ccccc2)OC)=O)CC(N=c2[nH]cnc3cnccc23)C1 89654,c1(C(=O)NC2CC(CNC(Cc3n(C)cnn3)=O)C2)ccc(F)cc1C(F)(F)F 89655,C12(N3CCN(c4cc(Br)ncn4)CC3)CCCCCC1NCC2 89656,Cc1cncc(C(=O)N(C2CN(C(=O)CC=CC(C)(C)C)CC23CC3)C)c1C 89657,C12(C(=O)NCC(=O)CCC3CC3(F)F)CCC(O1)c1ccccc12 89658,CCCC(O)CC(=O)NC(C)CNC(=O)COC(C)CC 89659,Cc1cc(CC(=O)NC23CC(C2)N(C(=O)CCn2cccn2)C3)cc(C)c1 89660,c1(OCC)ncc(S(=O)(=O)Nc2ccc(OCc3ccccc3)cc2)s1 89661,c1(C(C(N2CC(NC(CCS(C)=O)=O)C2)=O)C2CC2)cc(F)cc(F)c1 89662,C1(C(C)NC(c2ccc(CC)o2)=O)CN(c2nnc(C(C)(C)C)s2)CCO1 89663,C(=O)(C1=CCSC1)NCc1c(C(=O)NCCC(CC)C)cco1 89664,C(CC(C)C)(C(=O)N1CCC(c2ccc(C)nc2)C1)ONC(COCCOCC)=O 89665,C(C)(C(O)C(F)F)NC(c1cn(CCNC(C(CC)O)=O)nn1)=O 89666,C1(NC(C(C(C)OC)NC(=O)C=CCN2CCCC2)=O)CCN(C)C1(C)C 89667,C1(CNC(C2C(CC)C2)=O)CC(C)N(C(=O)C=Cc2cncs2)C1 89668,C(=O)(C(C)C(C)(C)O)NC1C(NC(c2c(C)[nH]c(C(C)(C)C)c2)=O)COC1 89669,N1(C(CCCCN(C)C)=O)CCC(NC(c2ccncc2Br)=O)C(O)C1 89670,C(=O)(CCC[N+](=O)[O-])N1CC(OC)(CNC(c2cnc(F)c(Cl)c2)=O)C1 89671,C#CC1(C(N2CCOC(COC)C2)=O)CN(C(=O)CC(F)(F)F)C1 89672,CC1(C(N2CCC(CF)(NC(c3coc4c3COC4)=O)C2)=O)CC2CCC1C2 89673,c1(C(C(=O)NCC(=O)OC)NC(=O)CCOCCOC(C)(C)C)cnn(C)c1 89674,c1(-c2ccn(CC)n2)nnc(SCCC(=O)O)n1-c1ccccc1C 89675,N1(C(c2c(C)cc(C)[nH]2)=O)CCC(NC(c2cnc(C(F)(F)F)nc2)=O)C12CC2 89676,N1(C(C2CC(C#N)C2)=O)CC(O)C(O)C1CNC(=O)CCc1cccc(Cl)c1Cl 89677,N1(C(CCc2onc(C)n2)=O)CCC(O)C(N(C(=O)C(C)OCCC(C)C)C)C1 89678,c1(C(=O)NCCC(C)NC(C=C(C)c2cccs2)=O)cnc(O)cc1C 89679,c1(C(=O)Nc2cc(OC)c(Br)cc2C)c(Cl)nc2cc(Cl)ccn12 89680,O=NN1CCCCC1C(=O)NC(CO)C(C)NC(C1(c2ccccc2Cl)CC1)=O 89681,C1(CC(=O)NC2(C)CC(NC(C(C)Cn3ccnc3)=O)C2)CCC(C)(C)C1 89682,N1(C(c2ccn(C3CCC3)c2)C(=O)NC(CC)(C)C)CCC(F)(CO)C1 89683,O=[N+]([O-])c1ccc(-c2cc(C3CC3)c(F)cc2F)c(Cl)c1 89684,N1(C(C)=O)CCC(c2cn(C(COC)CNC(CC)(C)CO)nn2)CC1 89685,C1(NC(=O)COC2COC2)CCC2CC1CN2C(C1CC1C(F)F)=O 89686,c1(CN(C(c2cccnc2)C(=O)OC)C)cc(Br)ccc1OC 89687,c1(C(=O)NCC(CO)NC(c2coc(C3CCC3)n2)=O)ccnc(C(F)(F)F)n1 89688,CCC(C)(C(=O)NCCOCCOCCNC(C)C(N1CCCCC1)=O)C(F)F 89689,C(=O)(CC(F)F)NCCOCCCN(C(=O)CCc1ncccn1)C 89690,c1(N2CCC(OC(C)C)C2)nc(C)cc(=NCCNC(=O)OC)[nH]1 89691,C(=O)(C1=CCN(C)C1)NC1CC(F)(c2cn(CCC(=O)OC)nn2)C1 89692,Cc1ccc(=N)[nH]c1C(N1CC(NC(=O)CC2CCC2)C2(CC2)C1)=O 89693,Cc1ccc(C(F)(F)F)cc1C(N1CCC(C)(NC(c2ccccc2)=O)C1)=O 89694,c1(C(N2CCCCC(CNC(c3ccc[nH]3)=O)C2)=O)ccc2c(=O)ccoc2c1 89695,[N-]=[N+]=NCCCCC(=O)NC1(C(=O)NCC2CCCC2O)CCC1 89696,C#CC1(C(=O)NC2COCC2CC=C)CCN(C(=O)C(C)S(N)(=O)=O)C1 89697,C#CC1(CO)COCCN1C(C1(CF)CC(F)(F)C1)=O 89698,c1(OC)ccc(CCC(=O)NC2CCC(NC(c3cnc(S)n3C)=O)C2)cc1F 89699,c1(N2CCC(CC=C)(COC)CC2)nc(=NC)[nH]c(=NC2COCC2F)[nH]1 89700,N1(C(c2c(C)cn(C)n2)=O)CCC12CN(C(c1cccc(C(F)(F)F)c1F)=O)C2 89701,Cc1noc(C)c1C(C)(C)C(=O)N(CCCNC(=O)C(C)NC(C)(C)C)C 89702,C(C(=O)NN1CCCC1C(=O)N(C)C(c1cnnn1C)C)OCC=C 89703,C1(NC(=O)Nc2c(OC(C)C#N)cc(F)cc2)CCCC2OCCC12 89704,C1(NC(CC2CC(C(=O)OCC)C2)=O)C=CCN(C(c2ccnc(C3CC3)c2)=O)C1 89705,C#Cc1ccc(C(=O)NC(Cc2ccco2)C(=O)NCCN2CCOC2=O)o1 89706,CN1CCOC(N(C(C(=O)NCCC#N)C(C2CC2)C2CC2)C)C1 89707,CC#CCC(C)N=c1[nH]c(=N)[nH]c(=NC(C)c2sc(SCC)nc2C)[nH]1 89708,c1(C(=O)NCCC2(OC)CN(C(C3CCC3CF)=O)C2)ccc(Cl)c(O)c1 89709,c1(CN=C(NCCOC)NCC2SCCc3ccccc32)ccc(S(N)(=O)=O)c(Cl)c1 89710,C1(CCC(=O)NCC(C)(C)F)CCN(C(c2cc(Cl)ncn2)=O)CC1 89711,CC1c2nnc(C3CC3)n2CCN1C(=O)NC(c1cncc(Br)c1)C1CC1 89712,c1(CC(=O)NCC(CNC(=O)C(CO)C2CCC2)OC)ccc(C(F)F)cc1 89713,Cc1ccc(SCC(=O)NC(C2CCCN2C(c2nccnc2Cl)=O)(C)C)cc1 89714,C(=O)(C(C)(C)CCCN=[N+]=[N-])N1C(CNC(C2(F)C(C)(C)C2(C)C)=O)CC2CC21 89715,CC1(C)COCCC1C(N1CC2CC2(NC(c2csc(-c3cnc[nH]3)n2)=O)C1)=O 89716,c1(CC(=O)NCCC(C)NC(C2CC3CCC2C3)=O)c[nH]c2ccccc2c1=O 89717,c1(C(C(=O)O)NC(CCn2cc(CCN(C)CC)nn2)=O)c(F)cccc1F 89718,C1(C(N2C(CNC(CC=CCC)=O)CC(C)(C)C2)=O)Cc2cncn2C(=O)N1 89719,c1(OC)cc(CC(=O)NCC(Cc2ccc(F)cc2F)C(N)=O)ccc1Br 89720,CCCCC(C)CCC(=O)N(CCCN(C(=O)CCc1c(F)cccc1F)C)C 89721,c1(C(=O)NC(CNC(=O)CCc2cscn2)CO)ccc2ccnn2c1 89722,Cc1coc(C(C)C)c1C(N1CCCCC1Cn1cc(C(=O)O)nn1)=O 89723,Cn1c(CNC(C2CCC(CNC(c3nccs3)=O)C2)=O)nnc1O 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89742,Cc1ncc(C(N2CCC2(C)C(=O)NC2CCCC(O)C2)=O)cn1 89743,C1(NC(C2(C)CC(=C)C2)=O)CC2CC(NC(=O)C=Cc3c(C)coc3C)CC12 89744,c1(NC(c2c(C)nc(C3CCCOC3)s2)=O)ncc(Cl)cc1C(N)=O 89745,Cc1ccc(CC(=O)NC(C)(CNC(=O)C(c2ccccc2)C2CC2)CO)cc1 89746,N1(C(c2cc(Br)cs2)=O)CCC2(CC2C(N2CCOCC23CC3)=O)C1 89747,C(=O)(CC(O)C(C)C)NC(COCC)C(=O)NCc1[nH]cnc1C 89748,C(=O)(C(F)(F)CF)NCCOC1CN(C(C(C)N(CC)CC)=O)C1 89749,N1(C(C(CC)F)=O)CCC(CNC(C2CCCS(=O)(=O)C2)=O)C1(C)C 89750,C(=O)(C1=C(C)OCCC1)N(CCNC(Cc1cccc(OC)n1)=O)C1CC1 89751,Cc1ccc(Br)cc1CN1CCCC(C(N2CCCC(C)(C)C2)=O)C1 89752,C(=O)(CCC(F)(F)C(F)F)N(C)CCC1CCN(C(=O)CC2CCOC2)CC1 89753,CCC(C(=O)NCc1n[nH]cc1C(N1CCC(CNCC)C1)=O)N(C)C 89754,CN1CCN(C(C2CC3(CCO2)CC3)=O)C(C(N2CCCC(C#N)C2)=O)C1 89755,C(=O)(C(C)(C)C1=CCN(C(c2cnc(OC)nc2)=O)C1)N1CCCC(CC)C1 89756,CCCC(C(=O)NCCN(C1CCCC1)C(c1ccsc1)=O)OC 89757,Cc1cnc2cc(C(N3CCN(C(C4CC=CC4)=O)C(CO)C3)=O)ccn12 89758,C#Cc1ccc(C(=O)NCC2(C)CN(C(=O)C(O)CC)CC2C)c(F)c1 89759,C1(N(C)C)CN(C(c2cc(F)ccc2NC(=O)NC2CCCC2)=O)CC12CC2 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89847,N12CCC3(CC1)CC3C2=O.N1(C(c2nc(CCC)sc2)=O)CCCC(C(C)=O)C1 89848,c1(C(N2CC(C)C(NC(c3cc(N)c(Cl)cn3)=O)C2)=O)ccc(C2CC2)nc1O 89849,O=C1CCN(CC(=O)Nc2cccc(Sc3ccc(Cl)c(Cl)c3)c2)C(=O)N1 89850,c1(CN2CCCC(C(N3C(C)COCC3)=O)CC2)ccc2c[nH]nc2c1 89851,C1(CC(N2CCC(CC(C)NC(=O)CSCCN(C)C)CC2)=O)CCC(C)(C)CO1 89852,O=C1Nc2cc(Br)cnc2C1=NOC1CC2CCCCN2C1 89853,CN1C(=O)CN(CC(=O)NCCC2(NC(=O)Cc3ccsn3)CCC2)C1=O 89854,C1(C(N2CC(NC(c3c(Cl)cn(CCC)n3)=O)C2)=O)CC2CCCC(C1)C2 89855,c1(C(N2CC(C3(NC(c4c(SC)ccs4)=O)CC3)C2)=O)c(C)ccc(C)c1O 89856,n1(CC(=O)NC2C(NC(C=CC(=O)OCC)=O)C2)cc(C(N)=O)c(O)nc1=O 89857,c1(N(C2CCN(C(c3c(OC)ccs3)=O)C2)CCO)nc(C)cc(C#N)n1 89858,c1(C(=O)NCCN(C(=O)C(C)(C)n2cnnn2)CC)cccc(S(C)(=O)=NC)c1 89859,C1(C#N)(C(=O)NC(C2(C(=O)N(CC(C)(O)CO)CCO)CC2)C)CC(=O)C1 89860,c1(N(C)C)nc(NC(C2(CNC(c3cc(Br)ncc3Br)=O)CC2)=O)cc(O)n1 89861,C1(=CC(N2CC3(N(C(C(C)CC4CCCO4)=O)CC3)C2)=O)CCCCCC1(F)F 89862,n1(CC)cc(S(=O)(=O)Oc2cccc(Nc3cc(C)cc(=O)o3)c2)cn1 89863,C=CCCCC(C(=O)NCCN(C)CCO)NC(c1ccccc1C#N)=O 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89935,c1(C(=O)NCC(C)N(C(C(C(C)C)NC(=O)OC)=O)C)cc(Cl)cc(Cl)c1 89936,c1(C(C)=O)cnncc1Br.c12ccccc1CC1CCN2C1 89937,C#CCC(O)C(=O)N1CC(C)(C(=O)N(C)Cc2cc(=O)cc[nH]2)C1 89938,C1(CNC(C(C(C)C)OCC)=O)CN(C)CCN1C(c1ccc(F)s1)=O 89939,Cc1ncc2n1CCC(C(=O)NCC1CCCN(S(C)(=O)=O)C1)C2 89940,Cn1ncc(C(N2CCC(C(F)C(N)=O)CC2)C(=O)NCCCC2CC2)c1Br 89941,C1(C(N(CC(F)F)CCC)=O)CCCC2(CCC2)O1 89942,N1(N2CCCC(C#N)C2)CCC2CC(NC(=O)CCc3nc(Cl)n[nH]3)C2C1 89943,C1(C(=O)NCC2CCC(NC(c3c(C)nns3)=O)C2)CC(c2ccncc2)=NO1 89944,c1(CCN=C(NCC(F)F)NCC2C3CCOCC23)cc(Cl)c2c(c1)OCCO2 89945,c1(OC)ncc(CN2CCCC(C(=O)N(CCO)CCO)CC2)cc1Br 89946,CCC1=NOC(NC(=O)N(CCCCc2ccccc2)C)C1 89947,Cc1cc(C(=O)NCC2(C(=O)NC(c3nncn3C)C)CC2)nc(C)c1 89948,C(=O)(CC(C)CC(C)C)NC(CCC)CC(=O)NCC1(OC)CCCC1 89949,c1(CCC(=O)NCC(CC)NC(C2CC(OC(C)(C)C)C2)=O)cccnc1 89950,CC1CC(NC(=O)CC2CSCCS2)CN(C(=O)CCN(C2CCCCC2)C)C1 89951,c1(OCC)ccc(F)c(C(N2CC(c3cn(CCN(C)C)nn3)C2)=O)c1F 89952,C#CC1(C(=O)NC2(C=C)CCCC2)CN(C(C2CCCN2C=O)=O)C1 89953,c1(C(N2C(CNC(CCSC)=O)CC2)=O)ccc(NCc2nc[nH]n2)cc1 89954,C1(N(C(=O)Cn2ccnn2)CCOC)CCN(C(=O)C(F)C2CCCC2)CC1 89955,C1(C)(C(N(CC(C)NC(Cc2ccc(C)cc2)=O)C)=O)CCCS1(=O)=O 89956,C(=O)(CCCCCN(C(=O)CCc1ccco1)C)NCC(CC(C)C)O 89957,c1(C(=O)NCC2CCN(C(C3ON=C(CC)C3)=O)C2)c(Cl)ccc2c[nH]nc12 89958,c1(C(=O)NC2CCC(N(C(=O)C3=C(Cl)CC3)C)C2)cc2n(n1)CCO2 89959,C1(CNC(C(C)(O)C2CCC2)=O)(NC(=O)CC2(O)CCCC2)CCC(F)(F)CC1 89960,c1(CCC)nc(C)c(C(=O)N(CC(O)CNC(=O)CCC(=O)OC)C)o1 89961,c1(C(N2CC(F)(CNC(c3n(CC)ncc3)=O)C2)=O)cn2ccn(C)c(=O)c2n1 89962,N1(C(=O)Nc2ccc3cnn(CCOC)c3c2)CCCC2CCNCC12 89963,C1(CNC(C(C)n2cccn2)=O)CCCC2(CN(c3ccc([N+](=O)[O-])cn3)C2)O1 89964,Cc1cc(F)c2cc(C(=O)N(C(C)CNC(C3CC(C)(F)C3)=O)C)[nH]c2c1 89965,C(CN=c1cc[nH]c(C(N)=O)n1)(c1ccc(F)cc1)NC(C)=O 89966,c1(C(=O)NC2C(CNC(C(C)(C)F)=O)CC2)ccc(Br)c(N)n1 89967,c1(C(=O)NC2CC(C)(NC(c3n(C)ncc3Cl)=O)C2)ncn2c1CCCCC2 89968,C1(NC(c2c(COC)ncs2)=O)(CO)CCN(C(C2CCCC2)=O)C1 89969,CCCCC(O)C(=O)N1CCN(C(c2cc(I)ccc2Br)=O)CC1 89970,C(C(=O)NCC1CN(CC(F)F)C1)(C1CCCC1)NC(=O)OC(C)(C)C 89971,C=CCC(C)(C)CC(=O)N1CC(CNC(C2CCN(C)C2=O)=O)OC(C)(C)C1 89972,Cc1ccccc1Cn1cc(CNC(c2cccnc2O)=O)nn1 89973,CCCCCC(O)CC(=O)NCC1CC1CNC(c1ccc(Cl)cc1O)=O 89974,CCC(C)CC(C(=O)NCC(C)(F)C(C)C)NC(=O)CCOCC1CC1 89975,Cc1cnc(C(=O)NCC(c2ccccc2)NC(C2COC(=O)O2)C2CC2)nc1 89976,N1(C(C(=O)N(C)C)=O)CCCC(C2CCN(C(C3(O)CCCCCC3)=O)CC2)C1 89977,C1(C(=O)NC(C(=O)N(C)CC)C)CCN(C(=O)c2c[nH]c(=N)c(C)c2)O1 89978,c1(C(NNC(=O)C2N(C(C)(C)C)CC2)=O)nc2ccccc2[nH]1 89979,C1(C(N2CC(C)(CC)OCC2)=O)CC2CCC(C1)N2C(=O)C(C)OC(C)=O 89980,c1(C(=O)NCC(CC(C)C)NC(=O)CC(C)F)cn2c(n1)CCC2 89981,C1(NC(c2c(CC)nns2)=O)CC2CN(C(=O)C(N3CSCSC3)C)CC2C1 89982,N1(C(COC)=O)CCC2(CC1)CC(NC(C13COCC1C3(F)F)=O)C2 89983,c1(C(=O)OCC)cnc(NC(c2sccc2NCc2ccc(F)cc2)=O)c(Br)c1 89984,C1(O)(CC#C)CC(C(=O)NCC2CCN(C(c3occc3C3CC3)=O)C2)C1 89985,C1(C(=O)NC2(CCC)CCNC2=O)CC(C)CN(C(=O)CC2CC(C)C2)C1 89986,c1(NCc2cccc(OCC)c2OC)c(C)ccn2ncnc12 89987,N1(C(C(C)OCCN(C)C)=O)CCC(CNC(=O)Cn2cc(C3CCOC3)cn2)C1 89988,Cc1nc(C(=O)NC2CN(C(=O)CCc3ccoc3)CCC2C)c2ccccn12 89989,CCCCCCC(C)CC(=O)NCCN(C(C1CCC2CC2CC1)=O)CC1CC1 89990,C(C(F)(F)C(F)(F)F)OCCC(=O)NCC(C1CCC1)C1CCC1.C1(=O)C(F)N1 89991,C=CCC(CC)C(=O)NC1(C)CCN(C(c2c(C)cccc2O)=O)C1 89992,c1(C(N(C2CCCN(C(C=Cc3occ(C)n3)=O)C2)C)=O)cccc(C)c1N 89993,C1(C(=O)NC(CNC(c2nc(O)c(C)s2)=O)CO)(COC)CCCCO1 89994,C1(C(=O)NC2C(NC(C(C)(C)OC)=O)CCCC2)CC2C=CC1CCC2 89995,Cc1ccc(SCC(=O)NCC(C)(O)CNC(c2ccccc2CO)=O)c(C)c1 89996,c1(C(=O)NC(C(C)NC(c2c(C)nccn2)=O)C)ncc([N+](=O)[O-])cc1Br 89997,C(=O)(CC(CC)C(=O)OC(C)(C)C)NC(CNC(C(CC=C)(C)C)=O)CC 89998,N1(C(C(C)(Cl)Cl)=O)CC2(C)CN(C(=O)C(O)C3CCCC3)CC2(C)C1 89999,O=C(C(O)CC(F)(F)F)OCCN(C(=O)CC(F)(F)F)Cc1ccccc1 90000,n1(CC)cc(CN(C(=O)C(CC2CCC2)NC(C2CCO2)=O)C)cn1 90001,c1(C(C2CCCC2)NC(=O)Nc2ccccn2)ccc(Br)c(F)n1 90002,c1(C(N(CCCNC(=O)CSC(F)(F)F)C)=O)cccc(N2CCCC2)n1 90003,c1(OC)ccc(NC(=O)C(C(C)CC2CCC2)N(CC(F)F)C)c(OC)c1 90004,c1(C(=O)NCC(CC)NC(C(C(=O)OCC)(C)C)=O)cc2ccc(C)cn2c1 90005,C1(NC(C2CC=CCO2)=O)CCCN(C(c2ccc(Cl)s2)=O)C1 90006,C1(CCNC(c2cnc(CC(C)C)[nH]2)=O)CCCN(C(=O)CCCC#N)CC1 90007,C(C(C)(C)CNC(C1CC1C)=O)N(C(=O)CNC(=O)NC)CC 90008,Cc1cc(C(=O)NCC2(C)CCN(C(c3cc(Cl)c(C)cn3)=O)C2)c(C)nc1C 90009,c1(C(=O)NCC(C)(CO)NC(c2cc(CO)ccn2)=O)cncc(Cl)c1 90010,Cc1cc(CC(=O)NC(CNC(=O)C(F)(F)C(O)C2CC2)C2CCC2)ccc1O 90011,c1(C(=O)NC2CC(N(C(C3C(C(C)C)CCC3)=O)C)C2)cnn(C)c1Br 90012,c1(C(=O)NCC2CCCCN2C(=O)CC2(C(F)(F)F)CCC2)ccnc(O)c1F 90013,C#CC1(C(=O)NCCC(C)(C)CC)CCN(C(C2CC3CCC3C2)=O)CC1 90014,n1(C(C)C)cccc1CNc1cnccn1.c1(C(C2CCCO2)(C)N)nnnn1C 90015,c1(CCCC(=O)NCC2CN(C(CC3(C)CC3(F)Cl)=O)C2)c[nH]c2ccccc12 90016,C(=O)(C(C)(C)CCCNC(=O)C(F)OC(F)(F)F)NC(c1ccc(OC)cc1)C 90017,c1(CC(N2CC(c3cn(C4(C)CC(C)(C)C4)nn3)C(O)C2)=O)ccnc2[nH]cnc12 90018,c1(CCCC(=O)N(C)CCNC(C2(C)CC2(F)F)=O)nc2ccccc2[nH]1 90019,Cn1ccc2sc(C(=O)NC3CC(NC(=O)C=CCN4CCCC4)C3)cc12 90020,N1(C(c2c(N(C)C)nccc2)=O)CC2(CCN2C(C2(C)CCCC2)=O)C1 90021,CCCCCCC(CC)NC1CC1C(=O)NC1(C(=O)NCC)CCC1 90022,Cc1nc(CO)sc1C(=O)NC1COCC1CNC(C1CC(=O)N(C)C1)=O 90023,C1(NC(CN(C)C)=O)COC2(CCN(C(=O)C(N)CN)CC2)C1 90024,N1(C(C2(C)CCC(C)CC2)=O)CCCC2CN(C(C3CC(=O)C3)=O)CCC12 90025,c1(N2CC3(CCN(C)C3)OCC2)nc2c(c(=NCC3CCCSC3)[nH]1)CCC2 90026,C(=O)(C1=CC2C=CC1C2)NC1C(CC(=O)N(c2ccc(Cl)cc2)C)CCCC1 90027,C1(C(C)NC(C2(C(=O)NC)CCC2)=O)CCN(C(=O)CCc2nncs2)C1 90028,N1(C(C2(CC(=O)OC)CC2)=O)CCC(O)(C(C)NC(=O)C(C2CCCCC2)F)C1 90029,c1(CC)nc(C#N)cc(=NCC2C(C)CCCN2C(c2cnnc(Cl)c2)=O)[nH]1 90030,C1(C(N2CC(C(N)=O)(CNC(C3CCC(CO)CC3)=O)C2)=O)CCCC(F)(F)C1 90031,N1(C(C2(SC)CC2)=O)CC(NC(=O)C(CC)c2ccccc2)CC2(CC2)C1 90032,N1(C(C(=O)NC)C)CC(O)(CNC(c2cn(CCC(C)C)nn2)=O)C1 90033,n1(CC)ccc(C(N2CCC(NC(=O)C(CC3CCCC3)OC)C2C)=O)c1C 90034,Cc1cc(C(C)C(N2CCC(Cn3cc(CCCO)nn3)C2)=O)c(C)o1 90035,CCCCC(CC)CC(=O)NCCCOCCNC(=O)C=Cc1cscn1 90036,C1(CC(N2CC(C)(NC(CC(CC)CC)=O)C2)=O)Cc2ccc(Cl)cc2C1=O 90037,c1(OCC)c(F)ccc(C)c1NC(C1(CNCc2ccccc2)CC1)=O.CN 90038,C12(CC(=O)NCCCCCC=C)CCC1CN(C(=O)Cn1ccc(C)c1)C2 90039,CCCCCCCC(=O)NC1CC(NC(=O)C(C)(C)C2CCCO2)CC1O 90040,CC1CC(=O)NCC1C(=O)NC1CCCC1CNC(=O)C=C1CN2CCC1CC2 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90058,Cc1cccc(Cl)c1CN1CCC(CO)C(C(=O)C(F)(F)F)C1 90059,C1(CNC(C(=O)N(CC=C(C)C)C2CC2)=O)CC(CO)CO1 90060,c1(CC)ccc(C(=O)NC(CNC(=O)CCc2cnn(C)c2)CC)cc1Cl 90061,c1(OC)cnccc1C(=O)NCc1csc(C(=O)NCC(C)(O)CCO)c1 90062,c1(C(N2CC(C)N(Cc3cccc4c3CCC4)CC2)=O)noc2ccc(Br)cc12 90063,N1(C(c2c(CC)c[nH]c2)=O)CC2CCCCC2(CNC(=O)CSCC(F)(F)F)C1 90064,C1(NC(c2csc(-c3cn[nH]c3)n2)=O)CN(C(c2cc(Cl)no2)=O)C2(CCC2)C1 90065,CC1CCc2onc(C(N3CC(O)C(O)C3CNC(=O)CSC(F)F)=O)c2C1 90066,N1(C(CCNC(COC)=O)=O)CC(N(C(=O)CC2CC=CCC2)C)C2(CC2)C1 90067,C1(C(N(CC(C)O)CCNC(c2cnsn2)=O)=O)CCn2c(O)nnc2C1 90068,C1(NC(c2n(C)ccn2)=O)CCN(C(C2OCC2(C)C)=O)C12CCC2 90069,CC(F)(F)CC(=O)NC1CC1NC(=O)COCc1ccncc1 90070,C1(NC(C(C)=C2CC2)=O)CCC(CNC(=O)C(C)Cc2cccnc2)C1 90071,c1(NCCn2cc(CNC(CC(CC)SC)=O)nn2)c(Br)c(C)nn1C(C)(C)C 90072,C1(CCC(=O)NC2CCOCC2NC(C2CC3(CSC3)C2)=O)CCC(=O)NC1 90073,C#CCC(C)(CC)C(=O)NC1CCN(C(c2ccc(O)c(C)c2C)=O)CC(O)C1 90074,N1(C(CCOCC(C)C)=O)CCCC(C2(NC(C3CCNC3=O)=O)CC2)C1 90075,S(=O)(=O)(c1ccc(=NCC2CCCCCC2(F)F)[nH]c1)N1CCC(=O)NCC1 90076,c1(C(N2CCC(N(C(CC=C=C)=O)CC3CC3)CC2)=O)cc(C)ncc1C 90077,c1(C(=O)NCC2N(C(CSCCC)=O)CC(F)C2)c(C)cc(OC)cc1F 90078,N1(C(C(c2ccccc2)OC)=O)CC(NC(c2cc(C)cc(C)c2)=O)CC(F)C1 90079,CCC(C(=O)N1CC2(CC(CNC(=O)CSC(F)F)C2)C1)C(F)(F)F 90080,c1(OC(=O)CCNCC2CCCN2CC2CCOC2)ccccc1Cl 90081,N1(C(c2c(C)nc(CO)s2)=O)CCC2CN(C(=O)Cn3ccccc3=O)CCC12 90082,CC1Cn2nc(C(N3CC4(CCN(C(C5CC5(C)Br)=O)C4)C3)=O)cc2C(=O)N1 90083,c1(C(=O)NC2CC(NC(CNS(C)(=O)=O)=O)C2)cccc(-c2ccccc2)c1O 90084,N1(C(C2(C)CCCN(S(CC(C)C)(=O)=O)C2)=O)C2CCC1CC(CO)C2 90085,N1(C(C(C)n2ccnn2)=O)C2CCC(C2)C1C(=O)NCC1(F)CCOCC1 90086,C(C(C(=O)NC(C)C)N1CCCC(c2ncc(C)s2)C1)(C1CC1)OC 90087,N1(C(C(C)OCC#C)=O)CCN(C(=O)C(C)OCC2(c3ccccc3)CC2)CC1 90088,N1(C(C)=O)CCN(C(=O)CN2CCN(Cc3ccc(I)cc3)CC2)CC1CO 90089,C1(N(C(CC)=O)C)CCCN(C(=O)Cc2cc(CC)no2)CC1 90090,N1(C(c2cc(CNC(c3[nH]cc(C)c3)=O)sc2)=O)CCC(C)(N(C)C)C1 90091,C1(C(N(C)CC2(NC(=O)CC3CCC(F)(F)C3)CC2)=O)CC2(C1)C(F)(F)C21CC1 90092,c1(C(N2CCC(C)(NC(C3CCC(CC)C3)=O)CC2)=O)[nH]nc2c1CCC2(C)C 90093,C1(CNC(=O)NC2CC(Cc3cnc(C(C)(C)C)o3)C2)Cc2ccccc2N1 90094,c1(CN2CC(C#N)N(C(c3ccccc3S)=O)CC2)ccc(F)c2ccoc12 90095,C(=O)(C(O)CCCNC(C1(C)SCCCS1)=O)N1CCN(CC(C)O)CC1 90096,Cc1cscc1NC(C1CCC(CNC(=O)CCc2cnn(C)c2)C1)=O 90097,C1(NC(CC(C)c2ccccc2)=O)CN(C(=O)CSc2nncs2)CC1C 90098,N1(C(COCCC#C)=O)CCN(C(=O)C(O)CC(C)C)C(c2ccccc2Cl)C1 90099,c1(C(=O)NCC2(C)CCN(C(C(C)(C)CC(F)F)=O)C2)cc(C#N)c(O)nc1N 90100,c1(C(CC)C)ccc(=NCCCOCCc2ccccc2)[nH]n1 90101,C(=O)(CCCC(F)(F)F)NCC(C1CC1)NC(=O)C=Cc1ccc(Br)s1 90102,c1(C(N2C(CNC(C3(CCOC)CC3)=O)CC2)=O)cc(C)c2c(c1)CCC2 90103,CN1CCN(C(C2CC23CCCCC3)=O)C(C(=O)NCC2CCC(=O)O2)C1 90104,Cc1cn2cc(C(=O)NCCOCCNC(c3ccn4ccnc4c3)=O)nc2s1 90105,N1(C(C(c2cccc(OC)c2)C)=O)CC2(CC(NC(=O)CCC(C)OC)C2)C1 90106,c1(C(=O)OC)nc(NC(c2cc(-c3ccc(Cl)cc3)[nH]n2)=O)cnc1C 90107,N1(C(c2c(C)noc2)=O)CCCC(C(N2CC=CC2CN(C)C)=O)C1 90108,c1(OC)nn(C)cc1C(=O)NCC1(NC(=O)C=CS(C)=O)CCOC1 90109,Cc1c(CC(N2CCOCC(C)C2)=O)sc2ccccc12 90110,C1(C)(CNCC(C2CCOCC2)NC(C2CC(C(=O)OC)C2)=O)CCCCCC1 90111,C(=O)(CC(C)CNC(C1CCS(=O)CC1)=O)N(C(C#C)C1CCC1)C 90112,c1(NCC2CCN(C(c3cc(C4CC4)ncn3)=O)C2)c(F)cccc1[N+](=O)[O-] 90113,Cc1ccc(C(=O)NCC(C)(Cn2cccn2)NC(=O)CCC2CC2(F)F)n1C 90114,c1(C(=O)OC)cc(C(=O)NCC2CN(C(=O)C(C)(C)SC)CCC2C)cc(F)c1 90115,c1(CC(=O)NC2C(NC(C(C)NC(C)=O)=O)COC2)csc2c(Cl)cccc12 90116,c1(NC(c2cccc(F)c2O)=O)ccc(-c2ccc(Cl)cc2C(=O)O)cc1F 90117,C(=O)(C1=NOC(C)(C)C1)N1C(CC(N(C)C[Si](C)(C)C)=O)CC(O)C1 90118,C1(N(CCC#C)CC2CCN(C(=O)C(O)CC#C)CC2)CCc2cnn(C)c2C1 90119,N1(C(CC2C3CN(C(c4n(CC)ccc4)=O)CC32)=O)CC=CC12CCOCC2 90120,C#CC1CCCCN1C(C1(C(C)NC(=O)C(=O)CC(C)C)CC1)=O 90121,c1(C(=O)NCCC2(C)CCN(C(COCCC=C)=O)C2)cccc2c1OC(C)C2 90122,C(=O)(C#CC(C)(C)O)N1C(C(=O)NC(c2ccncc2F)C)CC(OC)C1 90123,N12C(CC3CC13)C(=O)NCCC2=O.C(C(=O)N(C)CCOC)SCC 90124,c1(C(=O)NC(C2CC=CCC2)C(N2CCC(=C)C2)=O)cnc(O)cc1C 90125,c1(CC)nc(C)c(CC(=O)NC(C)(C)CCNC(=O)Cc2csc(C)c2)c(C)n1 90126,C1(NC(CCS(C)=O)=O)CCSC12CN(C(=O)CNC(c1ccc(N)cc1)=O)C2 90127,N1(C(CCc2cccc(C)c2)=O)CCCC(C(=O)NCC2CSCCO2)CC1 90128,C=CCCC(C(=O)NCC1(C2CC2)CCC1)NC(=O)CC1COC(=O)C1 90129,c1(C2(C(N3CCC(NC(C(COC)C)=O)C3)=O)CC2(C)C)cccc(Cl)c1 90130,C1(CNC(N(c2c(C)ccc(F)c2)C)=O)CCC2(CCCOC2)O1 90131,c1(C(=O)NC(C)CCCNC(C2CCC=CO2)=O)cnc2occc2c1 90132,N1(C(C(C(C)(C)C)OC)=O)CCC(C(=O)NCC(CC(C)C)N(C)C)C12CCC2 90133,C(C)(C(C)(C)C(=O)NC1CC2CCCC2C1)NC(C(C)C)=O 90134,Cc1cc(NC(=O)CCN2CCCC2)ccc1NC(C1CC(=C(F)F)C1)=O 90135,N1(C(c2cnc(Cl)s2)C(=O)NCCCC(=O)OCC)CCN(CC(C)O)C(C)C1 90136,CC(C)CC(C)CC(=O)N1CCCCC1CNC(c1cscc1C(N)=O)=O 90137,C1(CNC(C#CC(C)C)=O)CCCC12CCN(C(=O)CC1OCCC1C)CC2 90138,C1(NC(C2(SC)CC(O)C2)=O)CN(C(c2ccc(F)cc2)=O)C2(CCC2)C1 90139,N1(C(C(CC)C)=O)CC(CO)C2(C1)CN(C(=O)Cc1cccc(Cl)c1F)C2 90140,c1(-c2ccc(NCc3c(Br)ccc(C#N)c3)c(F)c2)cc2ccccc2cc1O 90141,CC(C)C(C(C)NC(=O)CCn1cncn1)NC(=O)Cc1ccc(O)cc1 90142,C1(C(C)NC(=O)C=Cc2ccco2)CN(C(=O)COCCF)CCO1 90143,CCC(C(=O)N(C(C)CCNC(c1ccc(S(N)(=O)=O)o1)=O)C)C(F)(F)F 90144,CN1CCC(OCC(=O)NCC2CN(C(=O)C(C)(C)c3cccs3)CCO2)CC1 90145,c1(C(N(CCCNC(C(C)c2cncs2)=O)CCO)=O)cc([N+](=O)[O-])ccn1 90146,C1(NC(C2(CC)CC2)=O)CC2(C1)CC(NC(=O)CCc1ccc(=N)[nH]c1)C2 90147,CN1CC(C(=O)NC(C)(C)C(=O)N(C)CCOC(C)=O)CCC1=O 90148,C1(C)(NC(Cn2nc(C)c(Cl)c2)=O)CCN(C(C2CCC(=O)N(C)C2)=O)CC1 90149,c1(-c2scc(Nc3nc(C)cc(OC)n3)n2)cc(F)c(Cl)cc1Cl 90150,N1(C(Cc2ccnc(OC)n2)=O)CCN(Cc2ccccc2)C(C(C)C)C1 90151,C1(NC(C2C(=C)CC2)=O)CN(C(c2cc3c(s2)CCC3)=O)CCC1C 90152,C1(CNC(=O)COC2CC2)COCCN(C(=O)CCOC2CCOC2)C1 90153,C1(Cc2c(C)cc(Cl)nc2)CCCCN1S(=O)(=O)N1CC(N)C1 90154,c1(C(N(CCN(C(c2c(C)noc2N)=O)C)C)=O)cc2c(F)c(F)c(F)cc2[nH]1 90155,CC1(C)CN(C(=O)CC2(O)CC2)C1C1CCN(C(C2CCS(=O)(=O)C2)=O)CC1 90156,c1(C(=O)NC(CCNC(C(CCC)C)=O)(C)CC)cc([N+](=O)[O-])c[nH]1 90157,S(=O)(=O)(c1cc2c(cc1Cl)CCCC(=O)N2)N1C(C)(COC)CC(N)C1 90158,CC(C)(C(=O)N1CCC(CNC(=O)C(C)(C)N2CCCC2)C1)C(F)F 90159,Cc1cc(F)sc1C(=O)NCC1(NC(C2CCC(C)O2)=O)CCCCC1 90160,Cc1cccc(C2CN(C(=O)C(c3ccncc3)C)C2)c1 90161,Cc1cc(=NCCCOc2ccc(O)cc2)[nH]c(C(F)(F)F)n1 90162,c1(CNCC(=O)NOC2CCOCC2)cccc(SC2CC2)c1 90163,c1(OC)ccc(-c2ccccc2)cc1CN(CC(O)C1CCC1)C 90164,C=CCC(CC(F)F)NC(=O)COC1CCN(C(C2(O)CCC2)=O)C1 90165,Cc1ccn2ncc(C(N3CCC4CC3CN4C(c3ccc(Cl)cc3)=O)=O)c2c1 90166,C(=O)(CCC(CF)CF)N1C(C)C(NC(=O)CN2CCOCC2=O)CCC1 90167,c1(NCCC(CNC(CCS(N)(=O)=O)=O)O)nc(Cl)[nH]c2nccc1-2 90168,C(C(CC(=O)NCCNC(N)=O)C1CCC1)NC(C(CC)N(C)C)=O 90169,C12(C(N(C3CC4(CC4)C3)C)=O)CCC(NC(C3CC4CCC4C3)=O)(CC1)C2 90170,C1(C(C)C)CN(C(=O)CC(C)(C)F)CCN1C(=O)CC1CCC(=O)N1 90171,Cc1cc(C(=O)N(C2CCN(C(c3ccc(C#N)cc3)=O)C2)CCO)ccc1Br 90172,C1(CNC(c2cnc(OC)s2)=O)CC2(CCN(C(C3SCCC3C)=O)CC2)C1 90173,N1(C(C2N(C(c3nnn(C)c3N)=O)CCC2)=O)CCn2nncc2C1 90174,N1(C(CCCCNC(C)=O)=O)CCCCC(C(N2CCCC(O)C2C)=O)C1 90175,c1(C(N(C)CC2(C)CCCC2NC(=O)C2=NOCC2)=O)cc2n(n1)CCNC2=O 90176,CCC(C)C(C)C(=O)NCC1(F)CC(NC(=O)CCc2ncc(F)cn2)C1 90177,CC(C)CC(O)C(=O)NC(C)CC1CN(C(=O)CCCn2ccccc2=O)C1 90178,C(=O)(CC(C(F)(F)F)NC(c1ccccc1F)=O)NCc1n(CC)ncc1 90179,N1(C(c2ccc(SCC)cc2)=O)CCC(F)(F)C(CNC(=O)CC(C)C)C1 90180,N1(C(CCOCCOC(C)(C)C)=O)CC=CC(NC(C2CCCN2C=O)=O)C1 90181,C1(C(=O)NC2C(CNC(C3(COC)CCCC3)=O)CC2)CCCS(=O)(=O)C1 90182,c1(C(N2C(CNC(C3C4CC5C(C4=O)C35)=O)CC2)=O)ccc2c(c1)CCOC2 90183,N1(C(C(C)NC(N)=O)=O)CC(F)(F)CC1CNC(C1(F)CCOCC1)=O 90184,c1(C(=O)NCC(C(C)(C)C)CO)cnc2cnc(Cl)cc2c1 90185,CC1(C)CN(C(=O)CCn2cccnc2=O)CC1NC(c1c[nH]cc(F)c1=O)=O 90186,c1(C(N2C(CNC(COCC=C)=O)COCC2)=O)cccc(C(N)=O)c1F 90187,c1(N2C(CNC(CS(CCOC)(=O)=O)=O)CCC2)cc2c(cn1)C(=O)CCC2 90188,N1(C(CNC(C)=O)=O)CC(c2ccccc2)(N)C1.C1(C(=O)N)CC1Br 90189,c1(C(N(CC(C)NC(=O)C(C)(C)c2ccns2)CC)=O)ccc(Br)cn1 90190,N1(C(c2[nH]nc(OC)c2Cl)=O)CCCN(C(c2ccc(C(C)O)cc2)=O)C(C)C1 90191,CCC(C)(CCNC(=O)Cc1ccccc1F)NC(=O)CC1CCCCO1 90192,Cc1ncc(CC(=O)NCC2CN(C(=O)CC3CNC(=O)C3)C2)c(O)n1 90193,C(=O)(C1=CCCC(C)(C)C1)NC(C1CCCN(C(c2ccc(SC)cc2)=O)C1)C 90194,N1(C(CCCC(=O)OC)=O)CC2CN(C(C3CCC(C)CC3)=O)CC2(C)C1 90195,c1(C(N)=O)cccc(N(C(C2CN3CCC23)=O)Cc2ccccc2)n1 90196,c1(C(N(CCNC(c2ccc(-n3ccnc3)nn2)=O)CC)=O)cc(Cl)nnc1O 90197,C1(NC(CCNC(C)=O)=O)CCN(C(=O)CCS(C)=O)C1C 90198,c1(OCCC)cccc(-c2cccc(OCC3(C)CC3)c2)c1 90199,CC(C)(C(=O)NC1CCC(CNC(C2(CO)CCCO2)=O)C1)S(C)(=O)=O 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90218,C1(CNc2c(OCCC)cccn2)CCCC2(CC(C(=O)O)C2)O1 90219,C1(C(CNC(COCCOC)=O)NC(C2CN(C)C2)=O)CCCCC1 90220,C(=O)(C1Cc2ccccc21)NCC(=C)CCNC(c1cccc(C)c1CC)=O 90221,CCC(C)CCC(=O)N1CCOC(CNC(c2ncoc2-c2cnn(C)c2)=O)C1 90222,Cc1nn(CCO)c(C)c1CNCCC(C)(O)c1ccccc1 90223,C(Cc1cnc[nH]1)(C(=O)N(CCO)CC1CC1)NC(=O)Cc1ccon1 90224,c1(C(N2CCC(C)C(NC(=O)C(C)(C)C)C2)=O)cc2c(nc1O)CCCC2=O 90225,C1(CC(=O)NC2(C)CN(C(C(C)CC3CC3)=O)C2)CCCC1(F)F 90226,Cc1cncc(C=CC(=O)NCCC2CCCCN2C(c2occc2C)=O)c1 90227,c1(C(N2CCCC(CNC(c3sccc3I)=O)C2)=O)cccc(F)c1I 90228,Cc1cc(C(=O)NCC(C)(C(C)C)NC(C2CC(CF)C2)=O)cc(C)c1O 90229,N1(C(c2c(OC)c[nH]n2)=O)CC2CC(O)C1C2NC(c1ccc2nnnn2c1)=O 90230,c1(NCCC(C=C)C)[nH]c(=NCCc2cccs2)nc2c1ncn2C(C)C 90231,C1(CCNC(c2n(CC)ncc2)=O)CN(C(c2snnc2C)=O)CCCO1 90232,c1(CNC(C2C(C)CN(C(=O)OC(C)(C)C)C2)=O)nc2ccc(Cl)c(F)c2[nH]1 90233,N1(C(C2(CN3CCCC3)CCCCC2)=O)CCC2(CCC(O)C2)C1 90234,N1(C(c2c(C)cnnc2)=O)CCC(C)(C)C(CNC(C2CCOC(C)(C)C2)=O)C1 90235,N1(C(C(COC)O)=O)CCC(C2CCN(C(=O)C(C)(C)C(C)(F)F)C2)CC1 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90254,C12(C(=O)NC3C(NC(C4CC5(CCC5)C4)=O)CCC3)CC3CC(CC1C3)C2 90255,c1(C(N2C(CNC(CN=S(C)(C)=O)=O)CC2)=O)cc(Cl)ccc1[N+](=O)[O-] 90256,C#CC1CC2(CC2)CN1C(=O)C(C)N(C(c1cc(C(C)=O)c[nH]1)=O)CC 90257,C1(NC(CCCCC(CO)NC(=O)OC(C)(C)C)=O)CS(=O)(=O)CC12CC2 90258,c1(C(=O)NCC2CCCC(NC(C3N(CC#C)CCC3)=O)C2)cc(Cl)nnc1Cl 90259,c1(COC)ccccc1CC(=O)N(C1CCC(NC(=O)Cc2cc(C)ns2)C1)C 90260,N1(C(C2CCC(=C)CC2)=O)CC2CCOCC2(NC(=O)CCC(C)C)C1 90261,C1(N(C(C(C)C)=O)C)CN(C(C2(CCN3CCCCC3)CC2)=O)CC12CC2 90262,C=CC(CCC)CC(=O)N1CC(N(C)C(c2ccc(F)cc2F)=O)C(O)C1 90263,c1(NC(=O)NCC2(O)C(SCC)CC2)nccc(C)c1N 90264,c1(C2C(NC(=O)NC(c3ccc(-c4cccnc4)cc3)C)C2)ccc(Br)cc1F 90265,N1(C(C=C(C)C(C)C)=O)CC(C(=O)NC(C)Cc2nc[nH]n2)C2(CC2)C1 90266,c1(C(=O)NCC2CC(NC(C3C(=C)CC3)=O)C2(C)C)ccc(C)c(C(F)(F)F)c1 90267,C=C(C)CCC(C)NC(=O)CC1CN(C(=O)CN2CCSCC2)CCO1 90268,c1(OCC)cc(N(C2CCN(C(=O)CC3CC(C)(C)CO3)CC2)C)ncn1 90269,CC(CN(C)C)C(=O)NC1CCCC1CNC(C1(c2cccs2)CC1)=O 90270,c1(OCC(N2CCC(Oc3ccc(C)cc3)C2)=O)c(F)cc(I)cc1F 90271,c1(NC2(CC=C)CCNCC2)nc(Cl)c(C)cc1C1CC(=O)Nc2ccccc21 90272,C1(NC(CC2(OC)CC2)=O)CCC2(CC1)CN(C(=O)CC1CCCC1)CCO2 90273,CCCCC(C)C(=O)NC1CCCCCC1C(N1CC[Si](C)(C)CC1)=O 90274,N1(C(CCC#C)=O)CCCCC(C(=O)NC2CC23CCCCC3)C1 90275,S(=O)(=O)(c1cccc2ccccc12)N1CC2CN(C(C3(F)CC3)=O)CC2C1 90276,C(CCC(CCC)NC(c1oc(SC)cc1C)=O)NC(CC(=C)C)=O 90277,N1(C(C(C)SC)=O)CC2(CCCCN2C(c2cnc3c(c2)CCCC3)=O)C1 90278,N1(C(CC(=O)NC)=O)CCCC(CC)C1C(N1CCCC(NC(C)=O)C1)=O 90279,N1(C(C(C2CN(C(c3c(OC)nccn3)=O)C2)O)=O)CCC12CCSCC2 90280,c1(NC(C)=O)ccc(C(C(=O)NCCC#N)N(C)CC2CCCCC2O)cn1 90281,c1(C2(C(=O)NOCCF)CC2)cn(CCCNC(N(C)C)=O)nn1 90282,C1(N(C)C(C2CC(F)(CF)C2)=O)CCCN(C(=O)COCCCF)C1 90283,c1(C(C(=O)NC(c2cnn(C)c2)C)O)ccc([N+](=O)[O-])cc1 90284,C(=O)(C(C)C1OCCc2sccc21)N1C(CC2CC(C(=O)OC)C2)CC1 90285,C1(CC)CN(C(C2(OC)CCOCC2)=O)CCN1C(c1occ2c1CCC2)=O 90286,CC1(NC(=O)CCc2cc(Cl)cc(Cl)c2)CCC(NC(C2CC(C)(O)C2)=O)CC1 90287,c1(CC(=O)NC2CC(NC(=O)Cc3cnc[nH]3)C2)csc2ccc(Cl)cc12 90288,c1(C(N2C(C)(CNC(c3cnc(C4CC4)[nH]3)=O)CCC2)=O)nc(Cl)ccc1N 90289,Cc1c(C(=O)NCC2(C(C)NC(C3CCCN(C)C3)=O)CC2)nnn1C(C)C 90290,Cc1c(C(=O)NCC=CCNC(c2ccc(Br)o2)=O)cncc1Br 90291,N1(C(c2c(C)nc(-c3ccccn3)s2)=O)CCC(C)C(NC(=O)C=CCF)C1 90292,c1(C(=O)NC2(C)CC(NC(C(CC)C(C)O)=O)C2)ccc2c(c1)CCCS2(=O)=O 90293,C1CCCCN1C(=O)CCNC(=O)CCN1CCCC1=O.C1(NC(C)=O)CCCC1 90294,C1(CNC(c2c(C)cno2)=O)N(C(C2CCS2(=O)=O)=O)CCC1(C)C 90295,N1(C(Cn2ccc(C)n2)=O)CC2(C1)C(NC(C1C=CCC1)=O)CCS2(=O)=O 90296,c1(C(=O)NC(CCCNC(C(C(C)C)OC)=O)(C)C)ncn2c1COCC2 90297,C1(CC(N2C(CC(=O)N(C3CCCOCC3)C)CCC2)=O)CCN(C)CC1 90298,C12(C(=O)NCCCCC3(NC(CCCC)=O)CC3)CCC(CC)(C1)OC2 90299,C(C1=NOC2OCCC12)Nc1ccc(CC(=O)NC(C)C)cc1 90300,C#CCC(C)(C(=O)N(CCCSC)C)NC(=O)C1=C(C)CCC1 90301,C1(NC(C(CC)N(C)C)=O)CCCCC12CCN(C(C1(C#N)CCCC1)=O)CC2 90302,C1(CNC(CC(=O)NCC#C)=O)COCCN(C(=O)CNC=O)C1 90303,c1(C(C(N2CC(NC(C3CC3(Cl)Cl)=O)C2)=O)F)ccc(F)cc1 90304,N1(C(C)=O)CC2(CCCC(CNC(c3cnsc3)=O)O2)C1 90305,c1(NC(c2ccc(OC3(C(N)=O)CC3)cc2)=O)ccnc(C(F)(F)F)c1F 90306,c1(NC2(c3ccc(-c4ccc(SC)cc4F)cc3)CC2)ncc2ccsc2n1 90307,C1(C(=O)NCCCOCCC(=O)NC2(CO)CC(OC)C2)C(C)(C)C1(C)C 90308,CCC(CC(=O)NCCC1(O)CCN(C(C2CN3CCCC2C3)=O)C1)C(C)(C)C 90309,CC1(C)COC(CC(N2CC(NC(c3cnc(C4OCCO4)s3)=O)C2)=O)C1 90310,c1(CC(=O)NCC2C3CN(C(C=C(C)C(F)F)=O)CC32)ccc([N+](=O)[O-])cc1F 90311,N1(C(C(CC)=CCCC)=O)CC2CC2C1C(N1CC(OCC(C)C)C1)=O 90312,c1(C(C)(C)C)nocc1C(=O)NC1CC(F)(CNC(c2ocnc2C(F)F)=O)C1 90313,CCCS(=O)(=O)CC(=O)NCC1(F)CCN(C(C2Cc3nccnc3C2)=O)CC1 90314,c1(OC)cccc(CC(=O)NC(C2(O)CCN(C(=O)CP(C)(C)=O)C2)C)c1Cl 90315,C(=O)(CCC(C)(C)C#N)NC1CC(C)N(C(=O)CSCc2ccccc2)C1 90316,C#CCC(C(=O)NN1CCCC1C(=O)N(CC)Cc1cn[nH]c1)OC 90317,N1(C(c2c(N)c(Br)cc(F)c2)=O)CCc2c(Cl)cccc21 90318,N1(C(C2(C)C(C)(C)C2CNC(=O)CSc2n[nH]c(=N)s2)=O)CCC2CCC12CO 90319,c1(CC)cccc(C(=O)NCC2=CCN(C(=O)C(N3CCC(C)C3)=O)CC2)c1F 90320,c1(C(=O)OCC)cnc(N2CCC(F)(CN(C)C)C2)nc1 90321,Cc1cc2c(cc1Cl)C(NC(c1ccc(NC(=O)NC3CCC3)c(Br)c1)=O)CO2 90322,C1(CC(=O)NCC2CC(OC)C2)CCN(C(c2cn(CCO)nn2)=O)C1(C)C 90323,Cc1ccc(C(=O)NC2CCCC(N(C(=O)Cn3cc(CO)nn3)C)C2)n1C 90324,C1(NC(=O)CCN2CCOCC2)CN(C(C2(c3cc[nH]n3)CCC2)=O)CC1O 90325,C1(C(=O)NCCCN(C(c2cnc(S)[nH]2)=O)C2CC2)(CO)CC(F)(F)C1 90326,Cc1nc(C(C)C)ncc1C(=O)N(C(C)CCNC(=O)C(F)=CCCF)C 90327,c1(C(N(CC(CC)NC(=O)Cc2sccc2Cl)C)=O)cnc(OC)cn1 90328,c1(C(C)=O)ccc(OCCO)cc1.c1(CN(CCC(N)=O)N2C(=O)C2)ccc(Cl)s1.OC 90329,C1(CC)(CC)CC(NC(=O)CC2CCC(=O)N2C)CN1C(=O)CCC1CCCC1 90330,S(=O)(=O)(c1ccsc1C(N1CCC(N(C)Cc2ccccc2)CC1)=O)NC 90331,CC1C(NC(=O)CCn2ccccc2=O)CCCN1C(c1ccc(C#N)s1)=O 90332,N1(C(C(C)NC(CC)=O)=O)CCN(C(C2CC3(C2)CC3(F)F)=O)CC1C 90333,Fc1ccc2scc(CNC3CCCCC3c3cccc(Cl)c3)c2c1 90334,C1(NC(CC2(C(=C)F)CCC2)=O)CC2CC(C1)N(C(=O)CCc1nc(C)no1)C2 90335,N1(C(c2cc(CC(C)C)on2)=O)CCCCC1CNC(=O)CCN1CCCC1 90336,c1(C(N2CC(CNC(=O)Cn3cc(C4CC4)cn3)C2)=O)cc(CC2CC2)ncn1 90337,CC#CCCC(=O)N1CCC(C(N2CC(C)C(F)C2)=O)CC1 90338,CC(C)CC(CNC(C1CCCCC(=O)N1)=O)C(=O)N(C)Cc1ccccc1F 90339,N1(C(c2c[nH]c(=N)s2)=O)CCC2(CCC(NC(=O)C3=CC4(CCOC4)C3)C2)CC1 90340,N1(C(C(C2CC2)OC)=O)CCC(NC(=O)C(C)(C)NS(C)(=O)=O)C(F)C1 90341,c1(CC)ccc(F)c(C(N2CC(NC(c3cn(C)nc3COC)=O)C2)=O)c1 90342,c1(C(=O)NCC2C(NC(C3(COC)CC3)=O)C2)cc2cnc(Cl)cc2s1 90343,C1(NC(=O)CSCc2ccc(Cl)cc2)CC2CC1N(C(c1cnco1)=O)C2 90344,c1(C(N2CC(O)(CCNC(c3nc(C#C)sc3)=O)C2)=O)nc(O)nc(O)c1N 90345,C1(C(=O)NCCC(C)(C)CNC(C2C=CCC(C(=O)O)C2)=O)(OC)CCCCC1 90346,N1(C(C)C)CCN(C(=NCC2CCCS(=O)(=O)C2)NCC2CCOC2)CC1=O 90347,c1(C(=O)NC)ccccc1OC1CCN(C(=O)NC2CC23CCC3)C1 90348,c1(OC)cc(C(C)CC(=O)N(C)CCN(C)C(N2CC3CC3C2)=O)ccc1C 90349,C(CCC(c1ccccc1)NC(=O)Cn1cc(CCCC#N)nn1)OCC 90350,c1(C(=O)NCC2CCN2C(C23CC(O)C2C3)=O)ccc2c[nH]nc2n1 90351,Cc1ncc(NC(=O)CC=CCNC(=O)C(C)CC2CC2)cc1Cl 90352,CS(=O)(=O)c1ccc(-c2nnc(C(=O)C(N)CCCc3ccccc3)o2)cc1 90353,C(CCC(O)C(=O)NCCN1CCOCC1C)NC(c1cc(C)oc1)=O 90354,C(=O)(CS(=O)(=O)N(C)C)N(CC(F)CNC(c1cnc(CC(C)(C)C)s1)=O)C 90355,C(C)(C)(CCCC(=O)NCc1cncs1)NC(CCc1ccn(C)c1)=O 90356,C1(CNC(CN(C)CC2CCCOC2c2cn[nH]c2)=O)CCCCC1NC(N)=O 90357,c1(CNC(=O)NCC2(CC)CCC2)cc(C(F)(F)F)ccc1Br 90358,C1(NC(C2CC=CCC2C)=O)(CO)CCN(OC)C1.c12cc(cs1)C(=O)NC2 90359,N1(c2ccc(C#N)cn2)CCC2(CCC(CNC(c3ccccc3)=O)OC2)CC1 90360,Cc1cc(C(N2CCOC(C(N3CCOCC3CN(C)C)=O)C2)=O)ccc1C#N 90361,N1(C(C=Cc2cncc(OC)c2)=O)CC2CCCC2(NC(=O)CS(N)(=O)=O)C1 90362,CCS(=O)(=O)c1ccc(F)c(C(=O)NCC2(F)CCC(NC(=O)C(O)CF)C2)c1 90363,CC1CC(C(=O)N2CCOCC2(c2ccc(F)cc2)c2ccccc2)=NO1 90364,c1(OC)cc(C(=O)NC(C)(CNC(c2ccc(C)cc2C)=O)C(C)C)c(F)cn1 90365,Cc1cccc(C(=O)NC(C)CCNC(=O)CCc2ccoc2)c1C(F)(F)F 90366,c1(C2N(C(c3nn(COC)cc3Br)C(=O)NC)CCC2)cc(OC)nc(Cl)c1 90367,C1(NC(c2ccc(C)c(C)n2)=O)CC2CC1CN(C(=O)C=CC(C)(C)C)C2 90368,C1(C#CC(=O)NC2CCN(C(=O)CNC(=O)NC3CC3)C(CC)C2)(CC)COC1 90369,C1(C(=O)CC2C(NC(c3ccc(-c4cc[nH]n4)s3)=O)CC2)CC(F)(F)C1 90370,CC1CCC(C)N(C(=O)CCOC2CN(C(c3cc[nH]c(=N)n3)=O)C2)C1 90371,c1(NC(C2C3CN(C(c4ncn5c4CCCC5)=O)CC23)=O)ccc2nccn2c1 90372,O=C1CN(CC2CC23CCC3)C(=O)N1CCCCn1cnnc1 90373,C(C(C)C(F)C(=O)N(C(CF)CF)C)NC(CCCC)=O 90374,c1(C(N2CC(CNC(c3cncc(C)c3)=O)C3C2C3)=O)coc2c1CS(=O)(=O)C2 90375,N12CCC(O)C(C1)C2=O.Cc1ccc(CS(=O)(=O)NCC2CCN(C)CC2)cc1 90376,c1(N2CCC(OC)C2)nccc(=NCCOC(=O)C=Cc2cccnc2)[nH]1 90377,C12CCN(C(C)C1)C(=O)C1(CCC1)Cc1cn2nn1.C1(OC)(CO)CN(C)C1 90378,C1(c2nc(C(C)OCC)nn2-c2ccc(Br)nc2)CCc2nncn2C1 90379,c1(C(=O)NC2(CF)CN(C(C(CSC)C)=O)C2)ccc2cncn2c1 90380,c1(C(C(=O)NCC(COC)C)NC(c2ccccc2)=O)cccc(OC)c1 90381,C12(CCN(C(=O)C(O)C(C)C)C1)C(=O)NC2.c1(CC)csnc1OC 90382,c1(C(=O)NCc2c(C(=O)NCC(C3CCCC3)C)occ2)cccc2cc[nH]c12 90383,CC#CC1CCN(C(=O)COC2CN(C(c3cc(CC)sn3)=O)C2)C1 90384,C1(NC(c2cnc(C(=O)OCC)s2)=O)CC(C)N(C(=O)CCSC2CCCC2)C1 90385,Cc1cc(C(N2CCC(CF)(NC(c3cnco3)=O)C2)=O)c2c(c1)CCC2 90386,N1(C(C2C(=C)C2)=O)CCOCC1CN(C(=O)CSc1n[nH]c(O)n1)C 90387,c1(OC)ccc(-c2cc(C(=O)NCc3ccc(Cl)c(F)c3)n[nH]2)c(F)n1 90388,C1(NC(C(C=C)O)=O)CCN(C(=O)C(C)NS(=O)(=O)CC)CC1(C)C 90389,C(=O)(C(C)(C)CC(=O)OC)NCCn1cc(C(N(C2CC(OCC)C2)C)=O)nn1 90390,c1(CCC(=O)NC(CCN(C(CCCCCC)=O)C)C)c[nH]c2c(C)cccc12 90391,C(C(F)C(=O)NCC1(F)CC(NC(=O)C(C)(C)c2cnco2)C1)N(CC)CC 90392,C1(CC)CCCC(CNCc2cc(Br)cs2)C1 90393,N1(C(C2(OCC(N3CCCC3)=O)CCCC2)=O)CCC(NC(CCOC)=O)CC1 90394,c1(NC2C(NC(C(C)(C)c3nccs3)=O)CCCC2)nc(O)c2cnn(C)c2n1 90395,C(=O)(C(C(C)C)NC(C1CCC(NC(C2(C(=O)OC)CC2)=O)CC1)=O)OC 90396,C(=O)(C(C)(C)CC(=O)NCC=CC(=O)NCCN1CCC(CO)C1)OC 90397,CC1(C)CCC(NC(C23CCC(CC2)C3)=O)C(NC(CC(=O)NCC2CC2)=O)C1 90398,S(=O)(=O)(c1ccc(S(=O)(=O)NCCC)cc1)N(CC(C)(C)N)CC#C 90399,C1(C(N2CCC(CCNC(c3c(OC)c[nH]n3)=O)C2)=O)CCN(C)CC1 90400,C1(C(N2CCCC(CC)(NC(c3cccn3C)=O)C2)=O)CCCC1P(C)(C)=O 90401,N1(C(C(F)OC)=O)CCc2ccccc2C1CNC(c1nccn1C)=O 90402,C1(C(=O)NC2C(CC(C)(C)C)C2)CCCN(C(C23CCC(CC2)C3)=O)C1 90403,N1(C(CC)=O)CCC2CCC(NC(c3cccc(Oc4cccnc4)c3)=O)C1C2 90404,C1(C(=O)NC(C(C)C)(C)CNC(c2cnc[nH]2)=O)CCC2(CCC2)CC1 90405,c1(CCC)ncoc1C(=O)NC(C(=O)N1CC(O)C1)C1(C)CC1 90406,Cc1cccnc1CC(=O)NC1(CC=CC(=O)NCCC2CCC3CC23)CCC1 90407,c1(CCC(N2CCCN(C(C(C)C)=O)CC2CO)=O)ccc2c(c1)COCC2 90408,CC1(C)C=C(C(=O)N2CC(CNC(C3(c4cc[nH]n4)CCC3)=O)CC2(C)C)C1 90409,c1(OCC)nc(N2CCN(C(c3cnn(C(C)C)c3)=O)CC2CCO)ncc1Cl 90410,C1(C)(CC)CCCN(c2ccc(C(N3CCC3(C)C(C)C)=O)nn2)C1 90411,C1(O)(CNC(=O)C(=O)NC2CC2)CCN(C(=O)C=CC(c2ccc(F)cc2)=O)C1 90412,Cc1cc(=O)ccn1CC(N1CC(F)CC1CNC(=O)CSCC(C)C)=O 90413,Cc1cc(C(N2CC(CC(C)NC(=O)Cn3cc[n+](C)c3)C2)=O)[nH]c1C 90414,C(CC(C)(C)CNC(c1ccc(-n2cncn2)nc1)=O)NC(c1c(C)csc1)=O 90415,C1(C)(C2CC(C(=O)NC(C(=O)Nc3cc(C)no3)C)C(O)C2)NC(=O)NC1=O 90416,C(=O)(C1=NN(C)C(=O)CC1)NC1CC2CC(NC(C3(OC)CCC3)=O)C1C2 90417,c1(C(N)=O)cc(=NCC2CCCCC2NC(C2CCCO2)=O)[nH]c(Cl)n1 90418,N1(C(CN(CC)CC)=O)CC2CC(O)C1C2NC(c1cn(C2CCCC2)nn1)=O 90419,C1(C(N2CCCC(CCC(N3CC(C)C(C)C3)=O)C2)=O)Cc2ccccc2C1 90420,N1(C(CCNC(=O)OC)=O)CC(CC(=O)N(CC(C)(C)N(C)C)C)CC1(C)C 90421,CCC(C)(O)C(=O)N1CC(CN2CCN(C(C3(S(N)(=O)=O)CC3)=O)CC2)C1 90422,N1(C(CCCCCC)=O)CC2(C1)CN(C(C1CCC1OC)=O)CC2CO 90423,CCC(C)CC(C)C(=O)NCCN(C)C(c1ccc(SCC)nc1)=O 90424,N1(C(COCC=C)=O)CC(NC(C2CC2CF)=O)C(C)C1 90425,N1(C(C(C)OC2COC2)=O)CCC(C)(C)C(CNC(c2ccc(=O)n(C)n2)=O)C1 90426,O=[N+]([O-])c1ccc(O)cc1CNCc1cc(Cl)c(F)cc1F 90427,c1(N2CCOCC(NC(CCNC(N)=O)=O)C2)ncc([N+](=O)[O-])cc1Br 90428,N1(C(C2(C#N)CCCC2)=O)CC(C2CN(C(C34CC(CO3)C4)=O)C2)C1 90429,c1(C(=O)NCC2(NC(C(CCSC)O)=O)CC2)c(C)ncnc1C 90430,N1(C(c2c(CC)con2)=O)CCN(C(=O)C(C)OCC(C)C)CC1CF 90431,c1(-c2nc(COCC)nn2C2CCCCC2C)ccn2c1CSCC2 90432,C1(C(=O)NCc2cn(C)cn2)(NC(C(C)c2cc[nH]n2)=O)CC1(C)C 90433,C1(C)(COC)CC(NC(c2c(Cl)cccc2Cl)=O)CN1C(=O)CCC(C)C 90434,C1(OC)CC(CNC(c2cn(C3CC3)nn2)=O)(NC(=O)C(C)C2CC2)C1 90435,n1(CC(=O)NC(CC(C)C)CNC(=O)CCCN(C)C)nnc2c1CCCC2 90436,Cc1ccc(C(C)C)cc1C(=O)N(C(C)CCNC(=O)C(c1cnn(C)c1)O)C 90437,CON(CCC(=O)N1CCN2C(=O)OCC2C1)C(=O)c1cccnc1F 90438,N1(C(C(COC)C)=O)CCN(C(=O)CNC(c2nccc(C)n2)=O)CC1 90439,N1(C(CC)=O)CCC(C(=O)NCC(c2cnn(C)c2)C)CC1C 90440,C1(C(N2CC(CCO)C(CO)C2)C(=O)NCC)CCC2(CCC2)O1 90441,c1(C(=O)NC(C2(C(=O)NC(C)(C)CCCF)CC2)C)ccc(C#N)cn1 90442,C=C1CCN(C(=O)CNC(=O)OCC)C(C(=O)OC(C)C(F)(F)F)C1 90443,c1(CC(=O)NC2CC(F)(CNC(=O)C(O)CF)C2)c[nH]c2cccc(F)c12 90444,c1(C(=O)NC(CCCNC(C(CC)N2CCCC2=O)=O)C)cnc(C(N)=O)cn1 90445,CC1OC(=O)NC1C(=O)NCCCC1CCCCN1C(c1cn(C2CC2)cn1)=O 90446,c1(CCC(N2C(C)CN(C(C3CC3(Cl)Cl)=O)CC2)=O)nc2cnccc2[nH]1 90447,c1(C(=O)NC(CN(C(=O)CCC2(C#N)CCC2)CC)C)cncc(C(N)=O)c1 90448,Cc1ncc(Br)cc1C(N1CC2C(NC(=O)CNC(C3CCC3)=O)C2C1)=O 90449,C12(C(=O)NCC3CCN(C)C3)CC(CO1)N(C(=O)CC1CCCC1)C2 90450,C1(CC)CCN(C(=O)C=CC2(C)COC2)C(C(=O)NCC2CCCC(C)(C)C2)C1 90451,C1(C(N(CC(C)NC(=O)CC2CNC(=O)C2)C)=O)CCC(=O)N(C)C1 90452,COn1cnc(C)c1C(N1CCN(CCNC(=O)Cc2cccnc2C)CC1)=O 90453,c1(C(C)C(=O)NC2CCCCC2NC(=O)CSCCC#N)cccc([N+](=O)[O-])c1 90454,C1(C(=O)NC(C2(C(N3C(CCC)CCC3)=O)CC2)C)CCOC(C)(C)C1 90455,c1(C(=O)NCCC2(O)CN(C(c3cc[nH]n3)=O)C2)c[nH]c2ncc(Br)cc12 90456,C(C1CCCCCC1)=CC(=O)N(C1CCN(c2nnc(C(N)=O)s2)C1)C 90457,c1(NCCC(C)S(C)=O)cc(=NCc2nc(C(C)(C)C)cs2)[nH]cn1 90458,C(=O)(CCC1=CCCCC1)N1CCC(C)(NC(=O)CC2CCC(=O)N2)CC1 90459,N1(C(CCN(C(C)C)C(C2CC(=O)CS2)=O)=O)CCCC(C(=O)NF)C1.N(C)C 90460,C1(NC(CCCC#C)=O)CCN(C(=O)CCc2ccc(Br)nc2)C(C)C1 90461,CN1CC2CCC(C1)N2C(C1CC(F)CN1C(=O)CC1CSCCO1)=O 90462,CP(C)(=O)c1cccc(C(=O)N=S2(=O)CCCCCC2)c1 90463,C1(NC(CC2N(C(C)C)CCC2)=O)(CO)CCN(C(=O)CCC2CC2(Cl)Cl)CC1 90464,c1(C(=O)NCC(CC=C)NC(=O)CCC(C)CC)nccc2[nH]nc(C(C)C)c12 90465,N1(C(C(CC)(C)CO)=O)CC23CCCC2(C1)CN(C(c1c[nH]cc(C)c1=O)=O)C3 90466,c1(CC)cc(C(=O)N(C(CNC(c2cn(C(C)C)cc2C)=O)C2CC2)C)nn1C 90467,C(=O)(C1=CCc2ccccc21)N1C(CNC(C2=CC(C)(C)C2)=O)C(C2CC2)CC1 90468,N1(C(c2c(C)nc(CC)o2)=O)CCC(C)(C)C1C(=O)NCC1CCCN(CC)C1 90469,C1(=CC(=O)NC2CC(F)(CNC(C3CCC(OC)C3)=O)C2)CCCCCC1(F)F 90470,N1(C(C(CCC)CC)=O)CC2(CCN(C(=O)C(c3cn(C)nc3C)C)C2)C1 90471,n12nc(C)c([N+](=O)[O-])c1N2CC.C1(C)CC(OC)C1.C(=O)(COC)OC 90472,N1(C(c2nc(C)nn2C)=O)CC(C)(CNC(=O)C=CC(F)(F)F)CC1(C)C 90473,CCCC(C)(C)C(=O)NCC(=O)NCC1(C)CCC(O)CC1 90474,C(=O)(C(C)(C)CCC#N)N1CC(CCNC(C(CC)N2CCCC2=O)=O)C(C)C1 90475,c1(C(=O)NCC(C)NC(=O)CC2CCC2(F)F)ncn2ccccc12 90476,c1(OCC)cnc(N2CCN(C(=O)Nc3cnn(CCCOC)c3)CC2)cn1 90477,c1(C(=O)NC2CN(C(=O)C=CCF)C3(CCC3)C2)c(Cl)nc2ccccn12 90478,CC1(C)CN(C(C2CC3CC3N2)=O)CCN1Cc1cc(Cl)c(Cl)c(Cl)c1 90479,N1(C(Cc2c(C)n[nH]c2)=O)CCC(NC(c2sc(CO)nc2C)=O)C1C 90480,CC#CCC(C)N=c1[nH]c(=NCC2(COC)CCCC2)[nH]c2c1CCCCC2 90481,C1(NC(C(CC#C)C)=O)CCC2(CC1)CN(C(=O)C(Cc1ccsc1)NC=O)C2 90482,c1(C(=O)NC(CN(C(c2ccc(CC)cn2)=O)C)C)ccnc(O)c1F 90483,C(=O)(C(C)(C)N=[N+]=[N-])N1CC(C=C)(CC(=O)NCC(C)OCC#C)C1 90484,CC1CC(NCc2nc(-c3ccccc3)n[nH]2)CN(C(=O)OC(C)(C)C)C1 90485,Cn1cc(N)c(C(=O)NCC2CN(C(C3CC3Cc3ccc(Br)cc3)=O)C2)n1 90486,C1(NC(c2cc(C(N)=O)[nH]n2)=O)CCC2(CCCN2C(=O)C2=CCCSC2)CC1 90487,C1(=O)C(C(C)(C)C)C2(CC2)N1.C1(n2cc(-c3cn(CC)nc3)nn2)CC2CCC1O2 90488,C(C(C)C(=O)N(CCNC(=O)Cc1sccc1Cl)Cc1ccccc1)OC 90489,c1(NC(CN2C(C(=O)OC)(CO)CCC2)=O)ccc(O)cc1O 90490,C(N=c1cc[nH]c(=NCCc2cncs2)[nH]1)C1(C)CC2CC2C1 90491,c1(CNC(N2CC(N3CCOCC3)CC2CO)=O)cnc(O)cc1O 90492,CC1Cc2cc(Br)ccc2N1C(c1cnc2c(c1)COCC2)=O 90493,N1(C(CC2CC(CC)OCC2)=O)C2CCC1C(CNC(C1CC1C(=O)OC)=O)C2 90494,N1(C(Cn2nc(C3CC3)n(C)c2=O)=O)CC(NC(C2CCO2)=O)C2CCCC2C1 90495,C(C(C)(C)C(=O)NC1CC2(C1)CC2C(N1CCC(F)(C(N)=O)C1)=O)OCC 90496,C(=O)(C1=CCC2(COC2)OC1)OCCc1c(C(=O)OCC)cccc1 90497,c1(C(=O)NC2C(NC(Cc3c(CC)cccc3)=O)CC2)cc(O)ccc1[N+](=O)[O-] 90498,C1(C(NN(CC)C(N)=O)=O)CCC2(CCCCC2)C1 90499,CCC(C)CC(C(=O)NC1CC(C)(CO)C1)NC(c1cncnc1)=O 90500,c1(C(=O)NCC23CC2CN(C(c2ccc(O)c(I)c2)=O)C3)cc(F)cc(F)c1F 90501,c1(C(=O)NCC(N(C(C(C)NC(C)=O)=O)C)C2CC2)nc(C2CC2)ncc1C 90502,N1(C(C2CCC(C(CC)(C)C)CC2)=O)CC2(C1)CN(C(c1nc(Cl)c(Cl)s1)=O)C2 90503,c1(NC(C(CC#C)NC(=O)C=Cc2ccncc2)=O)ccc(F)c(CC)c1 90504,C(CCC(=O)NCC(c1ccccc1)CNC(=O)C(=O)Nc1ccccn1)SC 90505,N1(C(C2(CC)CC2)=O)CCCCC1CNC(c1csc(NC(=O)C(C)(C)C)n1)=O 90506,c1(C(N(C(CNC(c2ncc(C)c(C)c2)=O)C)C)=O)cc(Br)c(O)nc1C 90507,C1(C2CCCN(C(=O)Cc3nncn3C)C2)(NC(C(C)OCCC(C)C)=O)CC1 90508,C(CCCCCN=c1[nH]cc(Br)cc1C#N)NC(C1(OCC)CCC1)=O 90509,c1(OC)ncccc1C(=O)NCCCCC1CCN(C(c2ccoc2)=O)CC1 90510,C1(NC(c2cc(CC)no2)=O)CC2(C1)CN(C(c1cc(Cl)cnc1O)=O)C2 90511,c1(OC)ccc(CN2CCC(O)(C(=O)NCC3CCC3)C2)c(Br)c1 90512,Cc1cc(=NCCCOc2ccccc2F)[nH]c(=NCc2cc(Br)cnc2O)[nH]1 90513,c1(C(=O)NC(CC)CNC(C2(S(C)(=O)=O)CCC2)=O)cnc(O)n(C)c1=O 90514,C1(C(=O)NC(C#C)CC(C)C)C2CCN(C(=O)CC(OCC)OCC)CC12 90515,S(=O)(=O)(c1ccc(NCc2c[nH]c(=N)s2)c(Cl)c1)NC(C(CCC)C)C 90516,N1(C(C=C(C)Cl)=O)CCC(NC(=O)CCn2c(C)csc2=O)CC(O)C1 90517,Cc1ccn2nc(C(N3CCCC(O)(CCNC(=O)C(F)(F)CO)C3)=O)nc2n1 90518,CC1(C)CCCCC1NC(=O)CCOCCCNC(c1nc(=N)cc[nH]1)=O 90519,c1(NC(=O)CC(C(F)F)NC(c2cn(C3CC3)nn2)=O)cccc2c1OCC2 90520,c1(C(=O)NC2C(CC)N(C(=O)CC3CC=CC3)CC2)cc2ccccc2c(=O)o1 90521,N1(C(Cn2c(C(F)F)cc(C)n2)=O)CC(NC(C2CC23CC(O)C3)=O)C(C)(C)C1 90522,C(N=c1cc(F)nc[nH]1)C1C2CN(C(C3C(c4ccc(OC)c(F)c4)C3)=O)CC21 90523,c1(-c2cccc(OC)c2)ccc2c(CC(=O)Nc3cn(C)nc3OC)n[nH]c2c1 90524,Cc1ccc(F)c(N)c1C(N1CC(CC(C)NC(C2CC2(F)Cl)=O)C1)=O 90525,Cc1nc(C(N2CC(C3(NC(=O)C(O)P(C)(C)=O)CC3)C2)=O)c2ccccn12 90526,C1(OCCNC(c2ccc(COC)s2)=O)CCN(C(=O)C(O)C(C)SC)CC1 90527,C12(CNC(CC3(C)CCCO3)=O)CC(CO1)N(C(C1CCCN1C=O)=O)C2 90528,O=S(=O)(C1CCC(c2ccccc2)CC1)NC1CCCCC1O 90529,S(=O)(=O)(c1ccc(NCC(O)CC(F)(F)F)c(F)c1)NC(c1csnn1)C 90530,C1(C(=O)NCC(C(C)C)NC(c2cccc(CCN(C)C)c2)=O)CC2(C1)CC2F 90531,C(=O)(CCP(C)(C)=O)N1CC(C)C(CCNC(C2(C(C)(C)O)CCC2)=O)C1 90532,C1(NC(CC2(NC(c3n(CC)ccc3)=O)CCC2)=O)CC2CCCCN2C1 90533,CCCCC(C)CCC(=O)NC1CC1NC(=O)CCc1cncn1C 90534,N1(C(C2CCN(C(C(COCC)C)=O)C2C(C)C)=O)CC2OC(=O)N(C)C2C1 90535,C12(NC(Cc3n(C)nnc3)=O)CCCC1CN(C(=O)CC1CCCSC1)C2 90536,C1(C(=O)NC2(CNC(c3ccc(CC)s3)=O)CCC2)CCCCC1F 90537,c1(-c2nc(CC(CC)C)nn2C2CC(c3ccccc3)C2)cccc2nc[nH]c12 90538,c1(CC(=O)N(CC(CNC(CS(CC)=O)=O)(C)O)C2CC2)cc(C)ccc1OC 90539,Cc1cc(Cl)c(C(=O)NC2CCCCN(C(=O)C(C)(C)C)C2)cc1C 90540,C(=O)(C(C(C)C)OC1CCCCC1)NCCCC(C)NC(CN(S(C)(=O)=O)C)=O 90541,C12(C(N3C(CC(=O)NCCc4ncc(C)o4)CC(F)C3)=O)CCC(C1)OC2C 90542,C(C1CCc2ncnn21)N(C)C(C1CCCN1S(=O)(=O)CCOC)=O 90543,c1(N2CCC(CN(C(=O)CCCn3c(O)nnc3O)CC)C2)ncnc(Cl)c1CO 90544,C1(C(=O)NCCC2(NC(C(CC=CC)C)=O)CC2)CC2(CCCCO2)C1 90545,c1(C(N(CC(=O)NCc2cccc(O)n2)CC2CC2)=O)ccc2cccnn12 90546,C(c1ccc(Cl)cc1F)=CC(=O)NC1CN(C(C(C(C)C)C#N)=O)CC1C 90547,CCCCC(CC(=O)N1CCCC1(C)COC)NC(c1c[nH]c(=NC)o1)=O 90548,C12(C(N3CCOCC(C(=O)NC4CCCC45CC5)C3)=O)CCC(CC1O)C2 90549,N1(C(c2c(C)nn[nH]2)=O)CC(N=c2[nH]c(Cl)nc3ccc(Cl)cc23)CC(C)(C)C1 90550,CN1CCC2(CCN(C(C3CCCC3CNC(c3cc(CCO)on3)=O)=O)C2)C1 90551,C(=O)(C(O)CC1CC1)NCC(C)=CC(=O)NC(CO)C1(O)CC1 90552,c1(C(=O)NC2CN(C(CCSC)=O)CC2C(F)F)cc(C)nc(C)c1 90553,C1(C(=O)NCC(CNC(=O)C=CSc2ccccc2)O)CCc2nnc(O)n2C1 90554,n1(CC)ncc2cc(C(=O)N(CCC(C)NC(=O)C(O)C(C)(C)C)C)c(C)nc12 90555,c1(CNC(=O)NC(c2c(SCC)cccn2)(C)C)cnc2ccnn2c1 90556,N1(c2cc(OC)ncn2)CC2(CN(C(C3CN(C4CCOC4)C3)=O)CC2CO)C1 90557,N1(C(c2ccc[n+]([O-])c2)=O)CCC2(CCC(C)C2)C1.C(C1C(=O)N1)OC(C)C 90558,c1(Cn2cc(NCC3CC(OCC(=O)OC)C3(C)C)nn2)sc(Br)c(C)c1C 90559,c1(C(=O)NC2C(NC(c3ccc(C(C)=O)cc3)=O)CC2)nccc2cnn(C)c12 90560,Cc1csc2ncnc(NCc3cn(C4CCC(C(=O)NCCO)CC4)nn3)c12 90561,C1(C(N2CC(CNC(C=C(C)C)=O)N(C)CC2)=O)CCC2(CC1)CC2(F)F 90562,N1(C(CCN(C)CC)=O)CC2CCC(N=C3N=CN[SH](C)C3)CC2C1 90563,CCC(C(=O)NCC(C)(C)CNC(=O)C=CCN(C)CC)OC 90564,Cc1cnc(N2CCN(c3cnn(C)c3)C(=O)C2)cc1C(F)(F)F 90565,c1ccc(N(C2CCCNC2)Cc2c[nH]nc2-c2ccccc2)cc1 90566,N12CC(C3CCCC13)C2=O.c1(OC)cncc(NC(=O)COC2CC=CC2)n1 90567,C(=O)(CC1=CCCCC1)NC(C)CN(C(=O)CCCCCc1cccc(O)c1)C 90568,c1(C(N2C(C(=O)Nc3c(C)ccc(F)c3)CC2)=O)ccc2n[nH]cc2c1 90569,c1(OC)cc(C(=O)N(C)CCOCCNC(=O)C(C)CCOC)cc(C)c1 90570,C1(CNC(c2ccc(CC)s2)=O)CCN(C(=O)C2=NNC(=O)C2)CC1C1CC1 90571,c1(C(NOCCC(C)C)=O)ccc(C2(NC(C3C=CCCC3)=O)CC2)o1 90572,C1(NC(C2(C)CC(=C)C2)=O)CCC2(CCCN(C(=O)C3=C(Cl)CCC3)C2)C1 90573,c1(OC(C)C)ccc(NC(=O)C(N2CCCC(C)(CO)C2)=O)cc1Br 90574,N1(C(c2n[nH]c(C)c2F)=O)CCN(C(c2coc(Cl)n2)=O)CC1c1ccncc1 90575,C(=O)(C1CCc2c[nH]nc21)NCCCC1CCN(C(C(C)CC2CC2)=O)CC1 90576,CCC(C#N)(CC)C(=O)N(CCCCN(C(=O)CN1CCCS1(=O)=O)C)C 90577,c1(C(C(=O)NC2C=CC(CNC(Cc3ccc(C)o3)=O)C2)C)ccncc1C 90578,CC1CCN(C(C2(C(F)F)CCC2)=O)CCN1C(C1C(c2ccccc2)C1F)=O 90579,C(=O)(C(O)CC(C)C)N(CCCN(C(c1sc(C)c(Br)c1)=O)C)C 90580,c1(N(C(c2c(C)nc(CC)nc2C)=O)C)cccc2cnccc12 90581,CC1c2ccccc2OC1C(N1CC2CC2(CNC(=O)CCC2CCCC2)C1)=O 90582,c1(C(=O)NCC2(COC)CCCN2C(=O)C(O)C2CC2)cnc(C)c(C(C)=O)c1 90583,C(=O)(C#CC(C)(C)C)NCCC(C)NC(C1(C)CCCC1(F)F)=O 90584,c1(C(=O)NC2C(C)CN(C(=O)COC3CC(F)(F)C3)CC2)cccc2c1CCC2 90585,c1(C(=O)NC2CC(C)(NC(=O)Cn3ncc(Br)n3)C2)cnc2ncccn12 90586,N1(C(CC=CCC)=O)CCCCC1CN(C)C(c1cc(C(=O)OC)nn1C)=O 90587,c1(C(=O)NCCc2ccc(COC)cc2)cnc(C)c(C#N)c1 90588,Cc1cc(C(N2CC(C)(NC(=O)CNc3ccccn3)C2)=O)ccc1O 90589,C1(C(=O)NC2C(SC)CN(C(=O)C(F)=C3CCCC3)C2)CC(C(C)C)=NO1 90590,C#CCCCC(C)C(=O)NCCn1cc(C(=O)NC2CCN(CC)CC2C)cn1 90591,CC1CN(C(c2cnc3[nH]nnc3c2)=O)CC(C)CN1C(=O)C1=CSCCO1 90592,N1(C(c2c(C)c[nH]n2)=O)CCOCC1CNC(c1csc(C(F)(F)F)c1)=O 90593,c1(C(C)NC(=O)C(C2CC2)NC(=O)CCCNC(N)=O)nccc(O)n1 90594,c1(CC)nc(C)oc1C(=O)N(CCC(=O)NC(c1ccccc1F)C)C(C)C 90595,c1(CCC(=O)N(C(CNC(C(CCC)C#N)=O)C)C)ccc2c(c1)OC(F)(F)O2 90596,c1(C(=O)NC2CCC(NC(CC=CCC)=O)CC2)cnc2c(c1)CCOC2 90597,CC(CCNC(=O)CCOCC(F)F)CCNC(c1c(Cl)csc1Cl)=O 90598,N1(C(=O)OC(C)(C)C)CCCC1CCN(C(=O)CCC1CCOC1)C1CC1 90599,c1(C(=O)OCCc2cc(OC)ncc2)ccc(C2CC2)c(Cl)c1 90600,C(C(CC(=O)NC(C)(C)CNC(c1cc(F)c(O)c(F)c1)=O)C(F)(F)F)N(C)C 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90936,c1(C(C(=O)NC2CC(F)(C(=O)OC)C2)C)cc(Br)ccc1C 90937,c1(CC(=O)NCCCOC(C)(C)C)ccnc(Cl)c1F 90938,N1(C(C2(C)N(C)CC(OC)C2)=O)C2CCC1CN(C(C1CN(C)C1)=O)C2 90939,c1(CCC)ccc(C(=O)N(CC(C)N(C)C(c2cc(C3CC3)nn2C)=O)C)cc1 90940,c1(N2CC(C(=O)OC)C(C(=O)O)C2)nc(C(F)(F)F)c(Cl)cc1Cl 90941,C1(=C(C(=O)N(C2CN(C(C3CC3F)=O)C2)C)F)CCCCC1 90942,C1(CN(C)C(C2CCNC2=O)=O)COCCN1C(c1ccc(C(F)F)s1)=O 90943,c1(C(CNC(=O)CCC2CCCO2)N(C(=O)C(F)=CCCF)C)ccccc1 90944,c1(C(=O)NC2CC(C)(NC(C=C(CC)C)=O)C2)cccc(C(C)=O)c1 90945,C(=O)(C#CC1CCCCC1)NC(C1CCCN1c1nnc(C2CCCC2)s1)(C)C 90946,N1(C(c2c(=N)cc[nH]c2)=O)CCOCC1CNC(C1CCC(F)CC1)=O 90947,c1(C(=O)NCC(CN(C(CCCC=C)=O)CC)(C)C)cc(C)nc2c1cnn2C 90948,CCCCC(C(=O)NCc1occc1C(=O)NC1CC2CCC(C1)N2C)C(C)C 90949,C1(C(N(C(CO)C2CC2)C)=O)CC(C)(C)CCN1C(c1csc(O)n1)=O 90950,CCCC(C)(O)CC(=O)NC(CCF)C(=O)N1CC(C)(CSC)C1 90951,Cc1cc(C2CC2)ccc1NC(=O)NC1CCN(c2cccc(Cl)c2)C1 90952,c1(C(CN(Cc2c[nH]nc2C)CC2CCC2)NC(C2C(CC)C2)=O)ccccc1 90953,C1(C(=O)NCc2c(CNC(CCC(=C)Cl)=O)nccc2)CCC2(CCC2)C1 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90971,N1(C2CC(n3cc(CCCCC(=O)OCC)nn3)C2)Cc2cnn(COC)c2C1 90972,C1(NC(C=C(C)C)=O)CCCC(NC(c2ccn(CC(F)(F)F)n2)=O)C1 90973,N1(Cc2cn(C(COCC)C(=O)NCCc3nnc(C)s3)nn2)CCOCC1=O 90974,C=CCC(C)C(=O)NC1CC(n2cc(CSCCO)nn2)C1 90975,C1(CC)CN(C(C2(c3ccccc3OC)CC2)=O)CCN1C(=O)Cn1nccn1 90976,c1(C(=O)NCCCN(CCCOC)C(C)C)ccc(Br)c(N)n1 90977,C(CC(C)C)(C(=O)NC1C(O)CC1O)NC(C(CCOC)OC)=O 90978,c1(C(N(C)CC2N(C(C(CCC)N(C)C)=O)CCOC2)=O)cccn2cncc12 90979,C(C)(C)(C(C)CC(=O)N)NC(c1c(CC)c[nH]n1)=O.C12(CC1)COC2.C(C)(C)O 90980,C1(Oc2ccc(Br)cc2)COC2(CCC2)C1.C12CN(C1)C(=O)COC(=O)N2CC 90981,CCCC(CC)CC(=O)N1CCC(C)C1CNC(c1c(C)nsc1C)=O 90982,N1(C(C2CNC(=O)O2)=O)CCC(CNC(C2(CC3CC3)CC2)=O)C(F)(F)C1 90983,c1(CC)ccc(F)c(C(=O)NC2CCCC2CNC(=O)C(C)C2=CCCC2)c1F 90984,c1(C(=O)NCC(C2CCCC2)NC(C(C)NS(C)(=O)=O)=O)nc2ncccn2n1 90985,Cc1noc(Cl)c1CCC(=O)NC1CCCN(C(C2CC2C(=O)NCCO)=O)C1 90986,N1(C(c2c(C)cns2)=O)CC(O)(C2(CNC(c3cc(F)cc(C)c3N)=O)CC2)C1 90987,CCCCC(CNC(c1ccc(C2CC2)s1)=O)NC(=O)Oc1cc(OC)ncn1 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91040,c1(C(N2C3CCN(C(CSC)=O)CC3CC2)=O)c[nH]c2c(F)c(F)ccc2c1=O 91041,S(=O)(=O)(c1cnccc1N1CCC(n2ccnn2)C1)NC1CCCS(=O)(=O)C1 91042,c1(C(=O)NCCN(C(=O)CC2(O)CCOCC2)C)ccc2ccncc2c1 91043,N1(C(CN(S(CC)(=O)=O)C)=O)CCC2CN(C(c3cc(C)c(N)cc3F)=O)C2C1 91044,C(=O)(C#CC1CCC1)NCC1C(CNC(c2c(OC(C)C)cccc2)=O)C1 91045,C(=O)(C1=CCCCC1C)NCCCN(C(c1cc(OC)c(Cl)cc1)=O)C1CC1 91046,c1(C(N2CCC(N(C(=O)Cn3cncc3C)CC#C)C2)=O)nccnc1CC 91047,N1(C(=O)CC2OCCO2)CCOCC(C(N2CC(n3cnnn3)C2)=O)C1 91048,C1(N(C(=O)Cc2n[nH]cc2Br)C)CN(C(=O)CNS(C)(=O)=O)CC12CC2 91049,c1(C(N2CC(O)C=C(C)C2)C2CCCC2)cnc2c(c1)c(C(F)(F)F)nn2C 91050,C1(C#CC(=O)NC(c2ccc(C)cc2)CNC(c2cc[nH]n2)=O)(CC)COC1 91051,C(C(C)(C)CC(=O)NC1CCCC1NC(c1cncc(N2CCCC2)c1)=O)OC 91052,C12(C(=O)NC3C(NC(c4nc(C)sc4)=O)C3)CCC(C(F)F)(CC1)CC2 91053,C(=O)(C1=CCC(C(F)(F)F)OC1)Nc1ncc(CCOC)s1 91054,N(C1CCOc2c(Br)cccc21)C(N1CCSC1CO)=O 91055,c1(C(N2CCC(C(C)C)(CNC(=O)CCC=CBr)C2)=O)cc2ccccc2n1C 91056,C1(OCCNC(CC2CC(OC)C2)=O)CCN(C(=O)Cc2ccnc(O)c2)CC1 91057,c1(C(N2CC(N(C(C(C3CCOC3)OC)=O)C)C2)=O)cnn(CC(F)F)c1 91058,N1(C(C(CC=C)C)=O)CC(C(C)(C)C)CC(CNC(C2(n3cccn3)CCC2)=O)C1 91059,CC1CN(C(=O)C=CC2CCOCC2)C(C)CN1C(=O)CCC(=O)OC(C)(C)C 91060,c1(C(=O)NC2C(CNC(=O)C=Cc3ccccn3)CCC2)cc2cccnc2s1 91061,CC1CCC(C)C1C(C)NC(=O)CC1CN(C(C2CC(CO)C2)=O)CC1C 91062,c1(C(=O)NCCC(C)N(C)C(c2ccn(C3CCC3)n2)=O)ccc(P(C)(C)=O)o1 91063,C(=O)(C(C)(C)CS(N)(=O)=O)N1CCCN(C(C2=CC(Cl)=C2C)=O)CC1C 91064,C1(CC(=O)NC)CN(C(=O)Cc2ccc(O)cn2)CCN1C(=O)CN(C)C 91065,N1(C(CCC(C)NC(c2n[nH]c(=N)[nH]2)=O)=O)C2CCC1CC(O)C2 91066,C1(O)(CN(C(C(CC)n2cccn2)=O)C)CCN(C(c2ncncc2N)=O)CC1 91067,CCCC(CNC(C1CN(C)CCO1)=O)C(=O)Nc1cnc(Cl)cc1C 91068,CCC(C)(C(=O)N1CCN(C(=O)C(=O)NCC(F)F)C(c2cn[nH]c2)C1)C(N)=O 91069,N1(c2n(CCOC)c(C3COC3)nn2)CCCC(C(C)C)CC1 91070,c1(C(N(C2CN(C(CCC=C)=O)CC2F)C)=O)ccc2nc(O)[nH]c2c1 91071,N1(C(Cn2c(C)ccc2C)=O)CC(NC(c2cc(Cl)sc2Cl)=O)CC(O)C1 91072,c1(OC)ccc(CN2CC3(CCN3C(=O)Cc3cc(C)n(C)n3)C2)cc1O 91073,C1(CNC(CCC2C(C)C2)=O)CCC2(CCN(C(c3cc(Cl)ns3)=O)CC2)O1 91074,Cc1c(CCC(=O)NC(CNC(=O)CN(C)C)C(C)C)c(O)nc2[nH]nc(O)c12 91075,c1(C(N(C2CCN(C(C34CCCC3C4)=O)C2)CC)=O)cnc2c(c1)CCC2 91076,c1(C2(C(N(C(CNC(c3nc(CCC)sc3)=O)C)C)=O)CC2)ccc(C)cc1 91077,C1(C)(C(=O)OC)C=CCN1C(C1OCCC1CNC(=O)Cc1cn[nH]c1)=O 91078,C1(C(=O)NC2CN(C(=O)NCC)C2)CCCCC1NC(=O)CC1CC(N(C)C)C1 91079,C1(C(C(=O)NCC(C2CC2)NC(c2ccncc2C(F)F)=O)F)CCCCCC1 91080,N1(C(c2c(C)csn2)=O)CC(C)CN(C(c2cnc(=N)[nH]c2)=O)CC1C 91081,C=CCC(C)(C)C(=O)NC1CCCN(C(c2ccc(CC)c(N)c2)=O)C1 91082,C(=O)(CCCC(=O)N1CC(NC(=O)COCP(C)(C)=O)CC1(C)COC)NCC 91083,C(=O)(CC(C)CCc1ccccc1)NC(CNC(C1CN(C(C)=O)C1)=O)(C)C(C)C 91084,N1(C(c2cccc3nncn23)=O)CC2CCC(C1CO)N2C(=O)C1=COCCO1 91085,C(CCC(CO)NC(=O)CC(C)(C)C)NC(c1scc(C)c1)=O 91086,c1(CC)onc(C)c1C(=O)NCCC1CCCCN1C(=O)CCNC(=O)OC 91087,CCCCC(CN=c1nc2cccc(Br)c2c[nH]1)NC(C1CC2CC2CC1C)=O 91088,N1(C(C2CCC(=C)CC2)=O)CCC2(CC1)CC(NC(=O)COC1(C)CCC1)CO2 91089,N#Cc1ccc(CCC(N2CC3C(NC(C4CCOC4)=O)C3C2)=O)c(F)c1 91090,c1(C(=O)OC)cc(I)cnc1NC(C1C2CC1N(c1cc(OC)ncn1)C2)=O 91091,CN(C)S(=O)(=O)N1CC(C(=O)NC2CC3(COC(CO)C3)C2)C1 91092,c1(CC)nc(C)c(C(N2CCC(C(=O)NCCC(C(C)C)OC)C2)=O)o1 91093,c1(C(N2C(CNC(C3CC4CC4C3)=O)CC(O)C2)=O)ncc(Cl)cc1Cl 91094,S(=O)(=O)(c1ccc(Cn2cc(C)cn2)cc1)N1C2CN(C(C(CC)=O)=O)CC21 91095,c1(SCC(=O)NC(C(C)C)C(C)NC(=O)C(C)(C)N(C)C)ncnc2[nH]cnc12 91096,CN=c1ccc(C(=O)NC2C3CC(NC(c4cnn(CC5CC5)c4)=O)CC23)c[nH]1 91097,C(CCCC(=O)NCC#CCNC(c1ccns1)=O)NC(N)=O 91098,c1(CC)c(C(=O)NC(C)CCCCNC(c2cnc[nH]2)=O)csc1C 91099,c1(C(=O)NCCC2(NC(C=C(C)Cl)=O)CCC2)ccc(C2CC2(F)F)cc1 91100,C1(C)(COC)CC(NC(=O)Cc2ccc(Cl)c(Cl)c2)CN1C(=O)CN(C)C 91101,c1(C2(NC(CCC3CCCC(=O)N3)=O)CCCC2)ccc2c(c1)OCCO2 91102,C=C(CNC(C1CCOC1CC)=O)CCNC(=O)C(C)OC(C)(C)C 91103,N1(C(C2C(C)(C(C)C)C2)=O)CCCC(NC(c2ccc(=O)n(O)c2)=O)C1C 91104,c1(C(=O)NCC(N(C)C(c2cocn2)=O)C2CC2)cccc(F)n1 91105,C1(NC(c2c(C)snn2)=O)CC2(CCN(C(c3sc4ccsc4c3C)=O)C2)C1 91106,C1(C(=O)NCCC(CC)C)CC2(CC2)CN1C(c1cc(C)sc1N)=O 91107,N1(C(C(CC)CN(C)C)=O)CCN(C(=O)COC2CC=CC2)CC1CCO 91108,c1(OC)ccnc(C(=O)N(CCCNC(c2c[nH]c(=N)o2)=O)C)c1C 91109,Cc1cc(OC2CN(C(=O)NCc3ccc(I)cc3C)C2)cc(C)c1 91110,c1(NC2(CC(=O)OC)CCOC2)ccc(C2(C(=O)O)CC2)cc1 91111,C1(NC(C2C(C)OCCC2)=O)CC2CCC1CN(C(c1cnccc1Cl)=O)C2 91112,C(C(C)(O)C1=CCC2CC1C2(C)C)NC(Cc1cn(C(C)C)nn1)=O 91113,C(=O)(CCCCC(N)=O)N1C2CC(CNC(C(C)CC3CC3)=O)C1CC2 91114,c1(OC)cc(F)ccc1C(=O)NCCC1CN(C(c2nc(C3CC3)oc2C)=O)C1 91115,N1(C(CC2C(C)CCN(C(=O)CCCC3CCCC3)C2)=O)C2CCCC1COC2 91116,C1(C(=O)NC(CNC(=O)Cc2cnoc2)C2CCC2)Cc2cccnc2C1 91117,Cc1ccc(C2CC2C(N2CCN(C(=O)CN3CCSCC3)CC2)=O)cc1 91118,N1(C(C2N(C(CC(C)C)=O)CCC2)=O)CCN(c2cncc(Cl)n2)CC1 91119,CCC(C)CC(=O)C(=O)NC(c1ccccc1)C(C)NC(c1cscc1Cl)=O 91120,C1(NC(CCc2cc(C)on2)=O)CC2CC(NC(=O)C=CCCC(C)C)CC2C1 91121,c1(C(=O)NCC(c2ccccc2)NC(C=CCN(C)CC)=O)ccc(N)cc1C 91122,C1(C(=O)NCC(C(=O)NCCNC(=O)NC)N(C)C)COCC1(C)C 91123,c12ncccc1NC2=O.C1(CN(C)C(N)=O)CCCN1C(=O)CSc1nncs1 91124,Cc1cc(OCC(=O)NCCC(C)CCNC(C2CC(C)(O)C2)=O)cc(C)c1 91125,C1(CC)CC(C(=O)Nc2cccc(C(F)(F)Br)n2)CCC1=O 91126,c1(C(N(C2C(C)CN(C(c3cn[nH]c3)=O)CC2)C)=O)cn(C)c2ccc(Cl)cc12 91127,c1(CCC(C)C)nc(-c2cnc(C3CCOCC3)o2)n(C2CCOCC2)n1 91128,CCCC(C(=O)NCC1CCCCN1C(=O)CC(C)(C)F)N(C)C 91129,c1(OCCNC(=O)Nc2ccc(SC)cc2)ccccc1OC1(CC)CCOC1 91130,C#CCCCC(C)C(=O)NC(C1(O)CN(C(c2ccsc2C)=O)C1)C 91131,C1(COC)(NC(=O)CCn2ccc(C)n2)CCN(C(C2CC(C#N)C2)=O)C1 91132,C1(C(=O)NCCNC(C2CCN(C3CC3)C2=O)=O)CCCc2ccccc2C1 91133,N#Cc1cc(F)c(C(N2CC(F)CC2C(=O)NCCC2CCC2)=O)c(Cl)c1 91134,CCC(F)C(=O)NC1CCC1NC(=O)Cn1cc(C(=O)N(C)C)nn1 91135,N1(C(C2C(=C)C2)=O)CCC2(CC1)CC(NC(C1CC3(C1)CC31CCC1)=O)CCO2 91136,C1(C(N2C(C)(C)CCC(C(=O)OCC)C2)=O)CCc2ncc(Br)n2C1 91137,C1(C(N2CC3CC2CN3C(=O)OC(C)(C)C)C(=O)NC)CC2OC(C)(C)OC2C1 91138,c1(C(=O)NCC(Cl)Cl)cc(CNC(c2cnn[nH]2)=O)cs1 91139,C1(C(=O)NCC2N(C(CNC(CCC)=O)=O)C3C(C2)C3)CCC(C)(F)CC1 91140,C1(C(=O)NCC(C)CNC(C2CC23CCC3)=O)CCc2ccccc2C1 91141,N1(C(Cc2c(C)noc2Cl)=O)CC(CO)C2(C1)CN(C(c1ccc(N)cn1)=O)C2 91142,C1(NC(CCSCC)=O)CN(C(=O)CSc2nncn2C2CC2)C2CC12 91143,C1(C)(COC)CCCN(C(=O)CN(C(=O)COC(C)(C)C)C)C1 91144,N1(C(C2C3C(NC(C(C(C)(C)O)(C)C)=O)C4C(C3)C42)=O)CCc2nnnn2CC1 91145,N1(C(C2=CC(O)C(NC(C(C)C3CC3)=O)C2)=O)CC2(C1)CC(C)(O)C2 91146,C(CC(O)C(=O)OC)NC(c1nnnn1Cc1cnnn1C)CCOCC=C 91147,C1(C(=O)NCC2(NC(c3cc(OC)ns3)=O)CC2)(COC)CCCO1 91148,N1(C(C2ON=C(C)C2C)=O)CCCC(C)(CNC(=O)C=CBr)C1 91149,c1(C(N2CC(CN(C(=O)Cc3ncc(Cl)s3)C)C2)=O)ccc(OC(F)(F)F)cc1 91150,Cn1cc(C(=O)NCC23CCC(C)(CC2)CC3)c(O)nc1=O 91151,N1(C(C(C2CCOCC2)C)=O)CCN(C(=O)CC2OCCO2)CC12CCC2 91152,N1(C(=O)C(F)CC2CCOC2)C2CCCC1CN(C(C13CCC(CC1F)C3)=O)C2 91153,C1(C(=O)NCC2(CNC(C(C)C(=O)N3CCOCC3)=O)CC2)CCS(=O)(=O)N1C 91154,N1(C(c2ccc(OCCCl)cc2)C(=O)NCCOC)CCCC(N=[N+]=[N-])C1 91155,CCC(C)C(C)C(=O)NC1CC(CNC(c2ccc(Br)c(O)n2)=O)C1 91156,N1(C(c2c(C)noc2)=O)CCCC(NC(c2nnc(C(F)(F)F)s2)=O)C1C 91157,c1(C(=O)NCCCC(C)NC(C2C(C)C2c2ccccc2)=O)cccnc1F 91158,C1(NC(=O)Cn2ccnn2)CCC(CCNC(C2(CCF)CCC2)=O)C1 91159,c1(CNC(C2CC=CC(NC(=O)CC3CCCC34CC4)C2)=O)cc(F)cc(F)c1 91160,C(=O)(CCN=C(NCC1(CC(N)=O)CCCCC1)NC1CC(O)C12CCC2)NC 91161,C(c1cccnc1)=C(C)C(=O)NC1CC1CNC(c1ccc(F)cc1)=O 91162,C1(C(=O)NC(CC=C)CNC(c2sc(F)cc2C)=O)CCC2CC2CC1 91163,CC1=C(C(=O)NCC2CCN2C(c2cc(Cl)ccc2Cl)=O)CCC1 91164,CC1(C)C(O)CCN1C(C1CCOCC1)C(=O)NCCC#N 91165,C#Cc1cccc(NNC(=O)Nc2cn3nccc3nc2C)c1 91166,N1(C(C2N(CC)CCCC2)=O)CCN(C(c2c(N)cc(Cl)cc2F)=O)CC(O)C1 91167,C(=O)(CCCS(C)(=O)=O)N1CCC(NC(c2c(C)n[nH]c2)=O)CC1C1CC1 91168,C1(NC(=O)Cc2cn[nH]c2)CN(C(c2ns[nH]c2=O)=O)CC(F)(F)C1 91169,N1(C(C(C)NC(CC)=O)=O)CCCC(N(C(=O)CSc2nncs2)CC)C1 91170,N1(C(c2c(C(C)C)nn(C)c2)=O)CC(NC(C2CC2C(F)F)=O)CC2(CC2)C1 91171,c1(OC)cnc2[nH]c(C(=O)NCC3(CNC(=O)C(O)C(C)C)CC3)cc2c1 91172,C1(NC(c2cn(C)nc2C(F)F)=O)CN(c2snc(Cl)c2C#N)C2(CCOCC2)C1 91173,c1(C(N(C2CN(c3cc(C)nn3C)C2)CCC)=O)cncc(-n2cccn2)n1 91174,C1(C)(CNC(C(CC)n2ccnc2)=O)CCN(C(C2CC3C=CC2C3)=O)CC1 91175,c1(C(N2CC(CCOC)N(C(=O)C3=C(C)CCC3)CC2)=O)c(C)cc(C)oc1=O 91176,c1(CC)ncc(C(=O)NCCN2CCCC2C)cn1 91177,C1(NC(CC2(NC(CCc3ncn(C)c3)=O)CC2)=O)CCS(=O)(=O)C1 91178,c1(C(C)=O)cccc(OCC(=O)NC2(CNC(C3CCCN3C)=O)CC2)c1 91179,C1(OC)CC(CCNC(=O)Cc2ccc(O)cc2)N(C(c2snc(O)c2Cl)=O)C1 91180,c1(C(CSCCC)(C)NCC2CC=CC2)nnnn1C(C)C 91181,C1(NC(C=CCNC(=O)CCOCC2CC2)=O)CC2(CCC2)C1O 91182,c1(CCC(N2CC(CCNC(=O)CCCF)OCC2)=O)nc2cc(Cl)ccc2s1 91183,Cc1ncc(C(N2CC3C(CNC(=O)Cc4ccns4)C3C2)=O)n1C 91184,c1(OC)cc(OC)cc(C(=O)NC2CC3CCC2N3C(=O)C(C)(C(C)C)OC)c1 91185,NS(=O)(=O)c1ccc(CC(=O)NC2(CO)CCCN(C(=O)C=C3CC3)C2)cc1 91186,N1(C(C2C(=C)C2)=O)CCC(CC)C1CNC(=O)COc1ccc(OC)cc1 91187,c1(SCC)cnccc1C(=O)N(CCCN(C)C(c1ccc(O)cn1)=O)C 91188,c1(CCNC(c2ncc(CCNC(C3C(C)C3)=O)s2)=O)c(F)cccc1Cl 91189,c1(-c2c(Cl)cccc2)nc2c[nH]c(=NCc3cnc4n3CCC4)nc2[nH]1 91190,N1(C(CCc2ccn(C)c2)=O)CC2CC(NC(=O)C3=CCCC3(C)C)CC2C1 91191,c1(C(C)=O)cc(C(N2CC(C(=O)NCC(F)CO)CC(F)C2)=O)ccc1O 91192,C1(NC(=O)CCc2cnoc2)CCN(C(=O)CN2CC3CC3C2)CC1O 91193,c1(OC)noc(C)c1C(=O)NCC1(C)CCN(C(=O)Cc2ccn(C(C)C)n2)C1 91194,C12(CC(=O)N(C(c3ccccc3)CNC(CSCC)=O)C)CCC(CC1)C2(C)C 91195,Cc1ccnc(C(=O)N(C)CC2(CNC(=O)CCn3cc(C)cn3)CC2)n1 91196,c1(C(N2CCN(C(C(Cc3ccccc3)OC)=O)CC2)=O)ccc(N)c(C)c1Cl 91197,c1(C(=O)NC2C(NC(C3(O)C(C)(C)C3)=O)CCC2)cccn2ncc(Br)c12 91198,C1(C(C)C)CCC(C(=O)NCC#CC2CC2)N1C(=O)CC1OCCCO1 91199,N1(C(C(C2CCCOC2)OC)=O)CCCC(C)(C)C1CNC(=O)C1=NOCC1 91200,C1(CNC(C(C)OC2CCCC2)=O)CCN(C(=O)Cc2ccc(F)nc2)CC1 91201,C1(CC(N2CCCC(N(C(=O)CCC3CC3)C)C2)=O)SC2=NCCN2C1=O 91202,c1(C(C)C)conc1C(=O)NCCC(C)NC(C1CCOC1C1CC1)=O 91203,c1(NC(C(c2cccc(Cl)c2)NC)=O)nc2cccc(Br)c2[nH]1 91204,C(=O)(CCCC(C)CC)NC(CC)C(=O)NCC1(C)CCC(C)CC1 91205,Cc1[nH]c2ccnn2c(=O)c1CC(=O)NC1CN(CC(F)(F)F)CC12CC2 91206,C=CCCC(C(=O)NC1(c2ccccc2)CC1)NC(=O)C(C(C)C)OCC=C 91207,c1(OC)ccc(COCCOC(=O)COc2ccc(O)cc2I)c(Cl)c1 91208,c1(OC)cncc(C=CC(N2CCC(NC(=O)Cc3ccoc3C)C2(C)C)=O)c1 91209,c1(CC)ccc(C(=O)NCC2CCC2NC(=O)C=CSc2ccccc2)c(O)c1 91210,c1(C(=O)NCCc2c[nH]c(=NCc3cc(F)cc(I)c3)s2)[nH]nc2ccncc12 91211,N1(C(CC2CCN(C)C2=O)=O)CC2(CNC(=O)CN3CCOCC3)CCC1C2 91212,CC(C)(CCC#N)C(=O)NCCC1CCC(NC(=O)Cc2ccoc2)C1 91213,Cc1coc(C)c1C(N1CC(CNC(=O)CCOCC(F)(F)F)C2CC12)=O 91214,c1(CNC(C(C)n2ccnc2)=O)cc(Cl)ccc1O 91215,N#Cc1ccc(F)cc1C(N1CCC(CNC(C2(Br)CC2)=O)CC1)=O 91216,Cc1cc(C)c(C(N2CCOC(C)(CNC(c3cnsn3)=O)C2)=O)c(C)n1 91217,N1(C(c2cncc(Cl)c2Cl)=O)CCC2(CC(NC(C3(O)CC3)=O)CO2)C1 91218,c1(C(C(=O)N(C2CCCCC2=O)C)C2CC2)ccc(Br)cc1 91219,C1(NC(C2C(C)C2C)=O)CCN(C(c2cn(C)[nH]c2=N)=O)CC12CCC2 91220,N1(C(C2(COC)CCOC2)=O)CCCCC(NC(c2ccc(C(N)=O)o2)=O)C1 91221,N1(C(CCC=C(C)C)=O)CCC2(C1)CN(C(=O)CC(C)Cc1ccccc1)C2 91222,CC1(C)CN(C(=NCC2CC3(CCC3)C2)NCc2cccs2)CCC1O 91223,Cc1cc(C(=O)NCCCNC(c2cc(C(F)F)ccc2F)=O)cc(N)c1O 91224,N1(C(c2[nH]n(C)c(=O)n2)=O)CC(F)(F)CC1CCNC(=O)CN1CCNC(=O)C1 91225,c1(CC)nc(C(=O)NCC2CC(O)CN2C(=O)C(O)CC)c(N)s1 91226,CC(C)CC(CNC(c1cnco1)=O)NC(=O)CCc1ccncc1 91227,N1(C(Cn2c(C)ccn2)=O)CCCC12CCC(NC(=O)C=Cc1cnc[nH]1)CC2 91228,CC1CCC(C(N2C3CCC2C(CNC(=O)CC2COC(C)(C)C2)C3)=O)CC1C 91229,C1(NC(=O)Cc2cnoc2)CCCN(C(=O)C(O)Cc2cnc[nH]2)C1 91230,C(=O)(C(C)(C)C(F)F)OC(C)C(N1CCCCC(CO)C1)=O 91231,c1(CC)occ(C)c1C(=O)NCC1CC1NC(C1CC1c1ccsc1)=O 91232,c1(N(C)C)cc(C(N2C3CCC2(CNC(c2ccns2)=O)CC3)=O)ccc1[N+](=O)[O-] 91233,N1(C(C)=O)CCc2cc(C(=O)NC3CC(C(=O)NC4(C)CC(C)=NO4)C3)ccc21 91234,c1(C(=O)NC(C(=O)N(CC(C2CCC2)OC)C)C)cncc(O)c1 91235,C1(NC(c2cnc(C(C)C)s2)=O)CN(C(=O)CC2CC(O)C2(C)C)CC1C 91236,c1(C(=O)Nc2c(Cl)ccnc2Cl)cn2c(n1)CN(C(C1CCOCC1)=O)CC2 91237,c1(C(N(CCCNC(C2COCC(C)O2)=O)CCO)=O)cc2cccn2c(O)n1 91238,c1(CNC(N2CCC(NS(=O)(=O)C3CC3)CC2)=O)ccc2nonc2c1 91239,c1(C(N2CC(C)C(NC(=O)C(CO)NC(N)=O)C2)=O)c[nH]c2c(F)cccc12 91240,C1(NC(c2c(C)sc(Cl)n2)=O)CCN(C(C2CN(C(=O)N(C)C)C2)=O)CC1F 91241,c1(OC)cc(C)cc(CN2CC3(CCC(C(=O)NCc4nccs4)O3)C2)c1C 91242,CCCCCCC(C)CC(=O)NC1CCN(CCCOc2cccc(F)c2)CC1 91243,C1(CNCc2cc(OC)c(OC)cc2)(CCCOC(=O)C(N)=O)CCCNS1(=O)=O 91244,C(=O)(CS(=O)(=O)CCO)NC(C)CN(C)C(C1(NS(C)(=O)=O)CCCCC1)=O 91245,CN1C(=O)Cc2c(C(=O)NCC(C3CCC3)NC(=O)Cc3cnns3)cccc21 91246,C(c1nc2ccccc2o1)=CC(=O)NC1C(CNC(C(C)(C)CO)=O)CCCC1 91247,CCCCC(CC)CC(=O)N1CC2(C1)SCCC2NC(c1ccc(Cl)nc1O)=O 91248,c1(OC)ccc(CC(O)C(=O)NC(CNC(c2cnc(O)o2)=O)C(C)(C)C)cc1 91249,C1(C(N2C(C(=O)OCC)CN(C(=O)C(F)(F)F)CC2)=O)CC(=O)CC12CCC2 91250,c1(-c2cc(C)no2)ccc(S(=O)(=O)N2CCCN(C(=O)C=CCN(C)C)CC2)s1 91251,C1(C(=O)OC)CN(C(=O)C(N2CCOC(CSC)C2)=O)CCN1C 91252,c1(C(N(CCCN(C)C(C2CC3(CC(=O)C3)C2)=O)C)=O)ccc(Cl)c(Cl)c1 91253,C1(NC(C=CCOC)=O)CCCC(NC(c2ccc(OC)nn2)=O)CC1 91254,CC(=Cn1ccnn1)C(=O)N(CCC(C)NC(=O)C(C)C1=CCCC1)C 91255,N1(C(CC2CC=C(C)CC2)=O)CCC(C(=O)N(c2cc(F)ccc2C)C)C(O)C1 91256,CC(C(=O)N1CCC(CN(C)C(c2cc(C(C)(C)C)nn2C)=O)C1)C(F)(F)F 91257,C#Cc1cncc(NC(C2(CNC(c3cc(C4CC4)no3)=O)CC=CC2)=O)c1 91258,N1(C(C(CC)NC(C)=O)=O)CC2CCC1C(CNC(C1(F)CCOC1)=O)C2 91259,O(C1CCc2c1cccc2[N+](=O)[O-])C(C1=NOC(C)C1)=O 91260,c1(CN2CCC(C(C(=O)NCC3CCCO3)OC)CC2)ccc(F)cc1C 91261,Cc1cc(C)n(CC(=O)N(CCCNC(=O)COCC2CCCCC2)C)c(=O)n1 91262,c1(OC)cccn2ncc(C(=O)NCC3(OC)CCN(C(c4ccsc4)=O)C3)c12 91263,N1(C(c2c[nH]nc2NC(=O)CCS)=O)CCCC(NC(=O)CC(C)C)C1.CO 91264,C1(CC=C)(C(=O)N(C)Cc2nc(C)ns2)CCCN1C(C1CC1C(C)(C)C)=O 91265,Cc1ccc(C#N)cc1C(=O)NC1CN(C(c2cc3n(c2)CCOC3)=O)CC1C 91266,C1(C(=O)NCCCNC(c2ccn(C3CCC3)n2)=O)CC2(CCCO2)C1 91267,c1(C(=O)NC(c2c(F)cccc2Cl)C(=O)OC)cc(Cl)ccc1Cl 91268,Cc1cccc(C)c1C(=O)N(CCC(C(C)C)NC(C1CCN1C(C)(C)C)=O)C 91269,C1(NC(c2c(SC)scc2)=O)CCN(C(c2[nH]nnc2C)=O)C(C)C1 91270,C1(NC(C=CC)=O)CN(C(=O)CCc2ccccc2N2CCOCC2)CC1(C)C 91271,c1(C(N2CCN(C(COCCCOC)=O)CC2C)=O)ccc(S(=O)C(C)C)cc1 91272,Cc1ccncc1C(N1CC(N(C)C)C(CNC(C2C=CCCC2)=O)C1)=O 91273,O=C(C1=C(c2ccccc2)SCCO1)NC1CCN(CC2(CC3CC3)CC2)C1 91274,N1(C(c2ncc(NC)nc2)=O)CC2CCC(N(C(=O)Cn3cc(Cl)cn3)C)C2C1 91275,Cc1cccc(C(=O)N(CCCNC(c2cnn(CC(F)F)c2)=O)C2CC2)n1 91276,C1(NC(=O)Cc2cc[nH]n2)CCCC(C(=O)NCc2nc(C(F)(F)F)cs2)C1 91277,C1(OC)CN(C(c2ccn(CCN(C)C)n2)=O)CC1NC(=O)C(=O)N(C)C 91278,C1(OC)(CF)CCN(C(=O)Cc2csc(C3CC3)n2)CC1 91279,C(=O)(C(O)CC1CCCO1)NCCOC(C)(C)CNC(=O)CCc1ncc[nH]1 91280,C1(NC(=O)C=Cc2cocn2)CC12CCN(C(c1cnn3c1CCCC3)=O)CC2 91281,O=C(CC1CC2(C1)CN(C(=O)CC1CCOC1=O)C2)Nn1cncn1 91282,C1(NC(C2COCCO2)=O)CCN(C(c2ncc(Cl)cc2Cl)=O)CC1F 91283,C1(CC)CCC(O)(C(=O)NCCNC(C2CN(C3(CC(=O)NC)CC3)C2)=O)C1 91284,c1(C(C)(C)C)ccc(NNC(=O)NCc2ccc(NC3CCOCC3)cc2)cc1 91285,C(CC1CCC1)(C(=O)N(C(C)C(=O)NCC(C)(C)O)C)OC 91286,c1(C(C)C(=O)NC2C3CCC(C3)C2(C)C)ccc(S(=O)(=O)N2CCCC2)cc1 91287,N1(C(CONC(=O)C2C(C(=O)OC)C2)=O)CCC(C2(C)CC2)C1 91288,N1(C(c2nnc(C(C)C)s2)=O)CCC(NC(=O)CCC2CC2(Cl)Cl)C(CO)CC1 91289,C1(C(C)NC(=O)C(C)(O)c2ccccn2)CCN(C(c2cccnc2)=O)CC1 91290,Cc1c(-n2nnnc2C(c2ccno2)NCC2CCC=CCCC2)cccc1Cl 91291,Cc1[nH]c(=N)ccc1C=CC(N1CC(C)(NC(C2CCN(C)C(=O)C2)=O)C1)=O 91292,c1(C(=O)Nc2c(C)c(Br)ccc2Br)cnc2c(C3=CCCCO3)cnn2c1 91293,C(=O)(CCC(=O)N(C)C)C12CC(NC(C(C)SC3CC(C)OC3=O)=O)(C1)C2 91294,Cc1cc(C(=O)NCCSCC(N2CCC(c3ncco3)C2)=O)nc(O)c1 91295,C(c1cc(C(N2CC3(CNC(=O)C(C)O)CC2CO3)=O)cc(OC)c1OC)=CC 91296,N1(C(CNC(CCCN(C(C)C)C)=O)=O)CCCCC1C(C)O 91297,CCC(C)CCCC(=O)NC1CN(C(c2ccc(C(=O)OC)cn2)=O)CC12CC2 91298,Cc1ccc(C(N2CCC(C(C)(C)NC(C3CCC(C(N)=O)CC3)=O)C2)=O)n1C 91299,c1(C(N(CC(CC)NC(=O)COC(c2ccn(C)c2)C)C)=O)ccc(OC)nc1 91300,C12(C(=O)NC3C(OC)CCC3)CC(CN(C(c3ccc(C4CC4)o3)=O)C1)C2 91301,c1(C(=O)NC2CC(C)N(C(=O)CCc3cnoc3)CC2)cccc2ccncc12 91302,C1(C2CCCN(c3nc(C)cc(C#N)n3)C2)(NC(C(CC(C)C)OC)=O)CC1 91303,N1(CC(=O)N(CC(O)C2(NC(c3cnn(CCF)c3)=O)CC2)C)C(=O)CNC1=O 91304,N1(C(c2c(C)ncs2)=O)CCC(c2ccccc2)(C(=O)NCc2cnn(C)c2F)C1 91305,N1(C(C)C)CC(NC(=O)C=CC2CCCN2C(C2C3CC4C(C3)C24)=O)C(C)C1 91306,C#Cc1ccc(C(=O)NC(C(=O)N(C(C)C(=O)OC)C)C(C)(C)C)cc1 91307,C1(C(=O)OC)CC2CC(C1)N(c1nnc(C(C)C)s1)C2 91308,Cc1sc(=O)n(CC(=O)NCC(C2CC2)NC(=O)CC2CCCS(=O)(=O)C2)c1C 91309,Cn1c(CC(=O)NCC2(F)CN(C(=O)CNC(=O)NC3CC3)C2)nnc1S 91310,c1(CC(N2CCCCC(NC(C(CCSC)O)=O)C2)=O)c(F)c(F)cc(F)c1F 91311,C1(NC(c2nn(CC)c(O)c2)=O)CC(NC(=O)C(C)(C)C2CCCC2)C12CCC2 91312,C(=O)(CCC(=O)c1ccccc1)N1CCC(CCNC(c2ccc(Cl)nc2)=O)C1 91313,N1(C(C(Cn2cccn2)NC(c2ccccc2F)=O)=O)CCCC2(CCCC2)C1 91314,c1(OCOC)cc(-c2nc(C(=O)Nc3cncc(C#N)n3)ccc2F)ccc1C 91315,Cc1cc(Nc2ccsc2C(=O)NC(c2ccccc2)CO)nc(Br)c1 91316,N1(C(=O)NCCOC(C(=C)C)=O)CCC2(CCN(Cc3cc(Br)ccc3C)C2)C1 91317,N1(C(Cc2cc(C)nn2C)=O)CCC(C(=O)NCCC2CCN(C)C2)=C(F)C1 91318,Cc1cn2c(C(N3CCC(CNC(c4sc(F)cc4C)=O)C(C)C3)=O)cnc2s1 91319,CC1CN(C(=O)CCc2nccn2C)CC1NC(c1cnncc1C(F)(F)F)=O 91320,c1(C(N(C2CCCCN(C(C(CCSC)O)=O)C2)C)=O)cc2n(c(=O)c1)CCS2 91321,C(N=c1cc(Cl)nc(C)[nH]1)C1N(C(C=CCOC)=O)CCCC1C 91322,N1(C(CCCC=C)=O)CC2CC(C1)C(CO)C2NC(=O)C(Br)=C(C)C 91323,C1(CC(=O)NCC2CC(NC(CC=CC)=O)C2)CCn2cncc2C1 91324,C1(C(N(CC(C)NC(c2cc(-c3ccccc3)cs2)=O)CC)=O)CC2(CCC2)C1 91325,C(=O)(CC(C)(C)C(=O)N1CC(OC)C(NC(=O)C(C)CC)C1)OCC 91326,Cc1nc(N(C)C)sc1C(=O)NCCC1CN(C(C2CC(C)(C)O2)=O)CCO1 91327,C1(=CC(=O)OC(c2ccccc2)COC)CCC(C)(C)CC1 91328,C1(N(C(CCc2cc(C)[nH]n2)=O)C)CN(C(=O)COCC2CCOCC2)CC1O 91329,CCC(C#N)(CC)C(=O)NCC1CN(C(=O)C(C2CCOCC2)O)C(C)(C)C1 91330,C1(C(=O)NC2(C(=O)OC)CC2)(NC(COCC=C)=O)CC(O)C1 91331,CP(C)(=O)C(CC(=O)NC1CCOCC1NC(=O)Cc1cncnc1)P(C)(C)=O 91332,C1(NC(Cc2n(C)ccc2)=O)CCC(C)(CNC(=O)CC2CC(=O)NC2=O)CC1 91333,N1(C(C2CC(NC(C3CC(CCC)C3)=O)C(O)C2)=O)CC2CC2C2CC12 91334,N1(C(c2c(C(C)C)noc2)=O)CC(C(=O)NCC2(C)CCCC2O)C(F)(F)C1 91335,c1(C(N2CCC(CN(C(=O)C=CC3CC3)C)C2)=O)ccc(Br)cn1 91336,N1(C(c2c(C)oc(C(C)C)n2)=O)CC(CNC(=O)C(=O)NCCC#N)CCC1C 91337,c1(N(C)CC2CC2(F)F)ncccc1S(=O)(=O)NC12CCC(C(F)(F)F)(CC1)CC2 91338,C(=O)(C(F)CC(C)(C)NC(=O)CCC1CC1(C)C)NCCSCC#C 91339,N1(C(C(CC)N(C)C)=O)CCC(O)(CCNC(c2[nH]c(C)nc2C)=O)C1 91340,C(CC(=O)N(C1CCN(C(c2nccc(Br)c2C)=O)C1)C)(C(F)(F)F)OC 91341,c1(OC)ccc2c(C(=O)NC3CC4CC3N(C(=O)Cn3cnnc3)C4)csc2c1 91342,CCC(C)C(C(=O)N(O)Cc1cn(-c2nccs2)nn1)Oc1ccc(F)cc1F 91343,C(=O)(CC(O)C(Cl)(Cl)Cl)NC(c1ccc(OC)cc1)CCCC 91344,c1(NC(C2(C)CCN(C(c3ccc(F)nc3F)=O)C2)=O)c[nH]c2ccc(Cl)cc12 91345,S(=O)(=O)(CC(=O)NCCCNC(=O)CC1OCCCO1)N(CC)CC 91346,CC1CC(NC(=O)Cc2ccc(OCC#N)cc2)CN1C(C1CCC(N(C)C)C1)=O 91347,C1(C(N2CC(=C)C2)=O)CC(C)N1C(=O)CC1(COC)CC1 91348,CCC(O)(CC(=O)NCC(C1CC1)NC(c1cncc(Cl)n1)=O)c1ccccc1 91349,C#CC1(C(=O)NC2CCC(CO)C2)CCN(C(C2CC3(CCC3O)C2)=O)C1 91350,c1(OCC=C)ccc(C(=O)NCC2CCCC2NC(c2nc(Cl)c(Cl)s2)=O)cc1 91351,C1(C(=O)NC(C)CCCNC(C2CCSCC2)=O)CCCC(C#N)C1 91352,Cc1sc(N)c(C(N2CCCC(CO)(CNC(=O)C(C)N(C)C)C2)=O)c1C 91353,C1(C)(NC(c2cc(SC)oc2)=O)CCN(C(=O)C(n2cnc(C#N)n2)C)CC1 91354,N1(C(c2ccc(CC)[nH]2)=O)CCC2(CC1)CN(C(=O)CC1CCC3CC13)CCO2 91355,c1(OC)ccc2c(c1)CC(OC)CN2C(=O)Nc1c(F)c(C)nn1C 91356,N1(C(CCN(C(C)=O)C)=O)CC(NC(c2nnc(S)n2C)=O)CC2(CC2)C1 91357,C(c1ccccc1)=C(CC)C(=O)NC1CCC(CCNC(C2(C)CC2(F)F)=O)C1 91358,Cn1cnc(C=CC(=O)NC2CC(F)(CNC(C3CCCC(F)C3)=O)C2)c1 91359,C(=O)(C1(C)CCc2ccccc21)NC1CN(C(C(C)(C)C2CC2)=O)CC1C(F)F 91360,CCCCCC(C)(C)C(=O)N(CC(C)CNC(=O)CC1CC(O)C1(C)C)C 91361,N1(C(CCCNC(C)=O)=O)CC(F)(F)CC1(C)CNC(=O)C(F)OC(F)(F)F 91362,N1(C(CSCCOC)=O)CCC(C)(CNC(=O)CN(c2ccccc2)C)C1 91363,c1(C(=O)NCC(CNC(C(C2CCCCCC2)C)=O)(C)C)cn(C)c(O)n1 91364,C#Cc1ccc(CC(=O)NC(CNC(c2cncc(C)n2)=O)CCCC)cc1 91365,N1(C(c2cc(CC)no2)=O)CCC(NC(=O)CCCF)C(C(N)=O)C1 91366,C(=O)(C(CCO)N(C)C)NC1CCC(NC(CC(=O)NCC)=O)C1 91367,C1(C(=O)NC2C(C)CN(C(c3coc(CO)c3)=O)C2)CN2CCC1(C)CC2 91368,c1(C(=O)NC2CCN(C(CC(CC)C)=O)CC2O)nc2ccccc2cc1Br 91369,C(=O)(CS(=O)(=O)C1CCCC1)N1CC(CCNC(C(C(CC)C)O)=O)OCCC1 91370,C(CC(C)C)(C(F)(F)F)NC(C(N1CCC(CNC(CCCC)=O)CC1)=O)=O 91371,C(=O)(CCCCCF)NCCNC(C1(SC)CCC1)=O 91372,c1(C(N(C)CC2C=CC(NC(=O)Cn3cccn3)C2)=O)cnc(C(C)(C)C)[nH]1 91373,N1(C(c2ccnc(C)n2)=O)CCN(C(=O)CC2CS(=O)(=O)C2)C2CC12 91374,C1(NC(C2CC(C)(c3ccccc3)C2)=O)COc2cc(-c3nn[nH]n3)nn2C1 91375,C1(CNC(C(C=C)O)=O)CCCCN(C(c2cc(=O)n(-c3ccccc3)[nH]2)=O)C1 91376,c1(SC)cc(C(=O)NC(CCNC(C2(C(F)F)CC(O)C2)=O)C(C)C)ccc1N 91377,N1(C(CNC(=O)OCC)=O)CCN(C(c2cccc(Cl)c2OC)=O)C(CCO)C1 91378,c1(CCC(=O)NC2CC3(C(NC(C(F)OC)=O)C3)C2)c(C)nc(O)nc1O 91379,c1(C(N2CCCC(Cn3cc(Cn4cncn4)nn3)C2)=O)cnc(C(=O)O)nc1 91380,N1(C(C2CC(=C)C2)=O)CC=CC1C(N1CCC(N2CCC2)C1)=O 91381,C1(NC(C(COC)C)=O)CCN(C(=O)Cc2ccc(OC)c(OC)c2)CC1O 91382,N1(C(c2c(C(=O)OC)c(C)[nH]n2)=O)CCCC(C)(NC(C2CC2(C)C)=O)C1 91383,CC(C)C1=CCC(C(N2C3CCC2CC(CCNC(=O)CSC2CC2)C3)=O)CC1 91384,N1(C(C(C)=C(CC)C)=O)CCC2(CCC2NC(C2COCCN2C=O)=O)CC1 91385,Cc1nccn1C(C)C(=O)NC1CCCC1NC(=O)CSCC(N)=O 91386,CN1CCn2ncc(C(=O)NCC3CN(C(=O)C(C)(C)C)CC3(F)F)c21 91387,c1(CC(N2C(CN(C(C(CC#C)C)=O)C)COCC2)=O)ccc(OC)cc1Cl 91388,c1(C(=O)NCc2nc(CNC(C(CC=C)OC)=O)sc2)c(C)[nH]c(C)c1C 91389,S(=O)(=O)(c1cncc(Br)c1)N1C(NC(c2cc(Br)nc(Br)c2)=O)COCC1 91390,C1(NC(c2ccc(C(C)=O)cc2)=O)(CO)CCCN(C(C2CC(O)C2)=O)C1 91391,C(C(C)(C)CC(=O)NCc1nnnn1C)NC(c1c(OC)nsc1)=O 91392,c1(C(N2CC(OCCNC(C3C(OCC)C3C)=O)C2)=O)cnnc(C)c1 91393,C1(C(=O)NCc2ncccn2)CC(F)CCN1C(c1cncc(Cl)c1)=O 91394,n1(CC)cnc(NC(=O)CCc2cc(C)no2)c1 91395,c1(CC)cc(C(=O)N(CCC(=O)N(CC)CC)C)no1.C1CC(=O)ON1 91396,c1(C(=O)NC(C(=O)NCCC(CC)O)C2(O)CCC2)c[nH]c2ccccc12 91397,c1(CNC(CN2CCN(C(C(CCC)NC(C)=O)=O)CC2)=O)ccc(Cl)c(Cl)c1 91398,C(=O)(C(C)C(C)NC(=O)COCCCOC)N(CC(=O)OC)CC=C 91399,CC(C)C(CC(=O)NC1(CCO)CCCCC1)NC(C1CCC2(CCC2)C1)=O 91400,N1(C(c2c(CC)cno2)=O)CCC(C)(C(=O)N(CC(C)C(F)(F)F)C)C1 91401,c1(CC(=O)NC2CN(C(=O)C3=CCCCC3)CC3CC23)ccc(F)cc1[N+](=O)[O-] 91402,N1(C(C2(CC#C)CCC2)=O)CCC(CO)(NC(=O)CCc2ccc(Cl)s2)C1 91403,CC1CN(C(C23CCC(CO)(CC2)C3)=O)CCC1NC(=O)Cc1cscn1 91404,C1(C(=O)Nc2ccnc(Cl)c2Br)Cc2cc(O)ccc2CN1Cc1cnc(Br)s1 91405,C(=O)(C#CC1CCCCC1)NC1C(NC(C(CCCC)CC)=O)COCC1 91406,C1(C(N(CC(COCC)O)C)=O)C2CN(C(C3(F)CC=CCC3)=O)CC12 91407,N1(C(C2(N(C)C)CCC2)=O)CCCC(C)(C(=O)NCCc2ccccn2)C1 91408,N1(C(CC(C)F)=O)C(CNC(c2cc(C3CCCC3)no2)=O)CC2CCCCC12 91409,N1(C(C2C(C)C2C)=O)CCC(C(C)C(=O)N(CCC(N)=O)C)C1 91410,c1(C(N2C(CNC(c3c(C)cno3)=O)CCCC2)=O)c(O)nnc2c1CCCC2 91411,Cc1ccc(CCC(=O)NC2CC2NC(c2c(C)noc2N)=O)cc1C 91412,C1(CNC(C=Cc2ccc(C)o2)=O)CN(C(c2cnnn2C)=O)C2CCCC2O1 91413,N1(C(COCCCCC)=O)CC2CCN(C(c3ccc(F)c(F)c3N)=O)C(C2)C1 91414,Cc1cc(=O)n(C)cc1C(=O)NCC1C(CNC(=O)C=CC2CCCN2C)C1(F)F 91415,c1(NC(C(C2CCN(C(C3C(C)(C)C3(C)C)=O)C2)F)=O)ccc(O)cc1F 91416,c1(NCC(N2CCN(OC)CC2)(C)C)ccc(S(=O)(=O)NC2CC2)cc1C#N 91417,c1(C(=O)NCCn2ccc(C(=O)NCc3nc(C)c(C)s3)c2)cn2c(n1)CCC2 91418,c1(CCNC(c2cc(Cl)ncc2Br)c2n(CCCF)nnn2)nnc2n1CCS2 91419,Cn1ncc(C(=O)NCc2occc2C(=O)NCC2CCCSC2)c1N 91420,c1(CN2CC(NC(=O)C=Cc3ccsc3)C2)cccc(C(=O)O)c1F 91421,C(=O)(C(C)CCCC(C)=O)NCC(C)=CC(=O)NC(C)Cn1cnnc1 91422,c1(C(=O)NC23C(CN(C(Cn4c(C)cnc4)=O)C2)CC3)nc2nccc(C)n2n1 91423,C(=O)(C1=CCCCC1C)NCc1ccc(C(N2CC=C(C)C2)=O)cn1 91424,C1(NC(C(c2n(C)ccc2)=O)=O)CCCC(NC(c2cnsn2)=O)C1 91425,C1(N(C)C(=O)NCC2CCN2C(=O)C=CSC)(C(=O)OC(C)(C)C)CCC(C)(C)C1 91426,Cc1cc(Br)c(CN2CCN(c3ccncn3)CC2C)cc1[N+](=O)[O-] 91427,C(=O)NN1CCC(F)(F)CC1.n1(CC)cc(C)c(C(C)(C)C)n1 91428,N1(C(C2CC(CC)C2)=O)CCCC(C2CN(C(=O)C=Cc3c(C)noc3C)C2)C1 91429,CC1CCC(CO)(NC(c2cncc(CNC(=O)C(C)OC(C)(C)C)c2)=O)C1 91430,C(=O)(C1Cc2ccccc21)NCC(CCNC(C1CC2(CC(=O)C2)C1)=O)O 91431,C1(CCC)(NC(C2CC3(CCC3)C2)=O)CCCN(C(C2CS(=O)C2)=O)C1 91432,N1(C(C(C2CCN(C(c3cc(C)c(C)[nH]3)=O)CC2)C)=O)CC2CCCC(C1)N2C 91433,c1(C(N2CC3CN(Cc4cnc(Br)c(F)c4)C3C2)=O)cc2cccc(Cl)c2[nH]1 91434,CC(C)C(C(=O)N1CCC(CCNC(=O)C(C)N(CC(F)(F)F)C)C1)C(C)C 91435,c1(C(=O)NC2CCN(C(C3C(C=C)CC3)=O)CC2CO)cccc2c1CCC2 91436,C(=O)(C1=CC2(CCOC2)C1)N1C2C(C(N(CC(CC)(F)F)C)=O)(CCC2)CC1 91437,c1(C(=O)OCc2cccc(F)n2)cc2ccc(Cl)cc2c(O)n1 91438,C1(C(N2CCCC(O)(CNc3ncc(F)cn3)C2)=O)CC2CCC1CC2 91439,C1(C(=O)NC(C)CNC(=O)Cc2cn(C)nc2Cl)CCc2nnc(O)cc2C1 91440,C1(CNC(c2ccc(CC(C)(C)O)s2)=O)CCCCN(C(C2CC=CCC2)=O)C1 91441,c1(NC(C(C)(O)C2CCCCC2)=O)cc[n+]([O-])cc1 91442,Cc1nc(C(=O)NCC(C(=O)O)C2CCOCC2)ccc1C#N 91443,N1(C(CC(C)O)=O)CC2(CCC(NC(=O)C=CCN3CCOCC3)CC2)C1 91444,C1(NC(c2cccnn2)=O)CCC2CN(C(=O)C=CC=C(Cl)Cl)CC2C1 91445,N1(C(C(CC)N(C(=O)C(F)(F)c2nccs2)CC)=O)CCCCC1COC(C)=O 91446,c1(C(=O)OC)ccc(C(N2CCCC2(C)C(=O)Nc2nnc(Br)s2)=O)cc1F 91447,Cc1cc(NC(C2CCN(C(c3cnn4cc[nH]c34)=O)C2)C)ncc1[N+](=O)[O-] 91448,C#CC1(C(=O)N(C)CC2CCCC2(C)C)CCN(C(=O)C(O)CC(F)(F)F)CC1 91449,c1(OC)cccc(C(N2CCCC2C(C(F)(F)F)NC(C2CC(C)(C)C2)=O)=O)n1 91450,c1(C(C)=O)cnc(N2CCCC(C(C)NC(c3cnc4sccn34)=O)C2)c(C)c1 91451,N1(C(C2CCCCO2)=O)CCNC(C(N2CCCC(F)C2)=O)C1 91452,N1(C(=O)OC(C)(C)C)CCc2ncc(NS(c3c(C)nn(C)c3C)(=O)=O)cc2C1 91453,C1(C(=O)NC2CCSC23CN(C(=O)CC(F)F)C3)CCCCC12OCCO2 91454,c1(C(N2CCOC(C(N3CC(F)(F)C(F)(F)C3)=O)C2)=O)cc2cc(F)ccc2[nH]1 91455,C1(C(N(C(C)(C)CC(N2CCC(F)CC2)=O)C)=O)CCCCC(=O)N1 91456,c1(NC(CNC(CC=CC=C)=O)C2CCC2)nc2c(C(=O)OCC)cccc2o1 91457,CN(C)NC(=O)CCC(=O)NCC1(C2CC2)CCN(C(C2(NC(N)=O)CC2)=O)C1 91458,c1(C(=O)NC(C(CO)NC(c2c(CC)scc2)=O)C)cc(F)cc2cc[nH]c12 91459,C(=O)(C(CC(C)C)C(C)C)NCCC(C(=O)NC1C(CCC)C1)OC 91460,c1(C(N(C)CC2OCCN(C(C3(C=C)CCC3)=O)C2)=O)cnn2cccc(Cl)c12 91461,C(=O)(CCCCCF)N(CC)CC1CCN(C(C2CN(C)CC2C)=O)CC1 91462,N1(C(c2c(-c3cn(C)nc3)c[nH]c2)=O)CCC(O)(CNC(C2CC23CC3)=O)CC1 91463,c1(C(=O)NC(CC=C)CNC(=O)C(C)CC2CC2)cnn2ccnc(C)c12 91464,C12(C(N(CC#C)C)=O)CCCC1N(C(CC(C)(C)C)=O)CC2 91465,C12(CNC(C(CC#C)C)=O)CC(CO1)N(C(=O)CC(C)(C)C=C)C2 91466,c1(OC)cccc(C)c1C(=O)NC(C)C(c1ccccc1)NC(C12CC(C1)C2)=O 91467,CCN=C(NCCc1cc(OC)cc(OC)c1)N1CCC(C(N2CCCC2)OC)C1 91468,C1(CNC(CCC=CC)=O)CCN(C(c2cnc(C(F)(F)F)s2)=O)CC1C 91469,N1(C(c2cc(C(=O)OCC)nn2C)=O)CCC2C(C1)CN2C(=O)CCC=CC(C)C 91470,Cc1ccc(Cl)c(OC(C)C(N2CCC(O)(CNC(=O)C(C)CC(C)C)C2)=O)c1 91471,c1(C(N2CCC(NC(C(CC)O)=O)CC2)=O)c(Br)sc(C)c1C 91472,n1(CC(N)=O)ccc(=NC(=O)C(CCC2CC2)NC(c2coc3c2COC3)=O)[nH]1 91473,N1(C(COCCCC)=O)CCCC(N(C(=O)C(C)NC2CCC2)C)C1 91474,C1(C(=O)NC(c2nncs2)C)CC12CCN(C(c1ccc(O)cn1)=O)C2 91475,C(CCC(C)C)(C(=O)NC1CCCN(C(=O)C(F)n2ccnc2)C1)NC(C)=O 91476,c1(C(=O)NC2CN(C(Cn3nc(C)oc3=O)=O)CC2(C)C)ccc2c(c1)CCC2 91477,C(=O)(C(CC(C)C)ONC(=O)CC1CC(F)C1)N(CC)CC1(O)CCC1 91478,C12(NC(COCC(=C)C)=O)CCCC1N(C(=O)Cc1ccc(O)cn1)CC2 91479,CCC(C)(CC)C(=O)NC1CN(C(=O)C(C)Cc2ccncc2)CC1OC 91480,c1(C(N2C(C)CC2(C)C)C(=O)NCCCF)ccc2c(c1)OC(F)(F)O2 91481,C(c1ccc(C(F)(F)F)c(O)c1)=CC(=O)NCC1N(C(CC(C)F)=O)CCC1 91482,N1(C(c2c(SC)cccn2)=O)CC(NC(c2csc(C)c2)=O)CCC1C 91483,c1(C)cc(C)c(C(=O)NC2CCCC2n2cc(CNC3CCOC3)nn2)o1 91484,c1(C(=O)NC2CCC2NC(C2CCCC2)=O)cnc2[nH]nnc2c1 91485,CCCCCCC(CC)C(=O)NC1CN(C(C2(NC(N)=O)CC2)=O)CCC1F 91486,c1(N(CCN(C(c2c(OCC)nc(C)cc2)=O)CC)CC)c([N+](=O)[O-])cnn1C 91487,CCCC(C#N)C(=O)NCC1(NC(=O)C=Cc2ccc(C(=O)N(C)C)cc2)CC1 91488,C1(C2CC2)(C(=O)NCC(c2ncn(C)c2)O)CN(C(=O)Cn2ncnn2)C1 91489,Cc1ccc(SCC(=O)NC2C=CCN(C(=O)COCc3nncn3C)C2)cc1 91490,c1(C(N2C(C(N(CC#C)CCF)=O)CC2C)=O)coc2c1COC2 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91578,c1(CNC2CN(C(c3n(C)cnc3)=O)CC2F)cc2c(Br)cccc2s1 91579,C(=O)(CCS(=O)(=O)c1ccc(C)cc1)N1CC2C(N(C(C(CC)O)=O)C)C2C1 91580,N1(C(C(CC)(F)F)=O)CCCOC(CNC(c2c(OC)ccnc2O)=O)C1 91581,C1(C)(C(N(CCCCN(C(=O)Cc2ccsc2Br)C)C)=O)CCCC1O 91582,N1(C(C(C)(C)NC(=O)NCC)=O)CCCC2(CCC(NC(=O)CCCOC)C2)C1 91583,c1(C(=O)NCC(C)N(C)C(C23CC2C3)=O)ccc(N)c(N)c1 91584,CCCCS(=O)(=O)CC(=O)N1CCCC2(CNC(C3(C(C)C)CC3)=O)CCCC12 91585,CCS(=O)(=O)c1cccnc1C(=O)NCC1(O)CN(C(C23COCC(C2)C3)=O)C1 91586,c1(CN(c2nnsc2C)CC(=O)NCC(C)(CO)NC(C)=O)ccccc1Cl 91587,C1(CC(=O)NC2C(CC(C)(C)C)C2)C2CCCC2N1C(c1ccc(C(N)=O)o1)=O 91588,N1(C(CNC(C)=O)=O)CCCC2(NC(=O)COc3ccc(C#N)cc3)CCCC12 91589,C1(CC(=O)NC2CC(OC)C2)CC(C)(C)CN1C(C1CCCOC1)=O 91590,c1(NC(=O)NCC2COC3CCCC3O2)c(C(F)(F)F)nc2n1CCCC2 91591,N1(C(C=CCOC)=O)CC(NC(C2CCN(C(=O)OC(C)(C)C)C2)=O)C(O)C1 91592,C#CC1(C(=O)NCCOCCOCCOC)CN(C(=O)C(O)CCN(C)C)C1 91593,Cc1cc(C)c(C(=O)NCC2CCCCN2C(=O)C(c2ccnn2C)O)o1 91594,C(=O)(C(CC(C)(C)C#N)N1CCN(C)CC(O)C1)NCCCCCC 91595,CC(C)(C(=O)NC1CN(C(c2ncc(Cl)cc2Cl)=O)C(C)(C)C1)C(N)=O 91596,C1(NC(C2C(C(C)C)C2)=O)CN(C(=O)C2=CC(C)C2)C2CCCC12 91597,c1(CNC(C2(OCC)CC2)=O)cc(C(=O)NCCSCCO)no1 91598,C1(C(CNC(CC2N(CC)CCC2)=O)(C)C)CCCCN1C(=O)COC 91599,CC1CCN(C(c2cc3ccsc3[nH]2)=O)CCN1C(=O)C=C1CCSCC1 91600,c1(C(N2C(C)CCC(NC(C3CC(C)(C)CN3C)=O)C2)=O)cc(F)cc(N)c1F 91601,c1(C(N(C2CCN(C(C3CC3COC)=O)CC2)CC#C)=O)cccc2sccc12 91602,c1(OC)c(C(=O)NC2CC(NC(C3CCCC3O)=O)C2)cc([N+](=O)[O-])cc1Cl 91603,c1(OC)ccccc1C=CC(=O)NC1CCCCC1N(C(=O)CSC(F)F)C 91604,CCC(CC)C(C)C(=O)N(C)CC1CCCN(C(C23CCCN2CCC3)=O)C1 91605,Cc1ccc2c(C(=O)N(C(C)CCNC(=O)C(CN(C)C)C(C)C)C)csc2c1 91606,C1(COC)CCCC(N(CCCNC(C2(CC3CC3)CC2)=O)C2CC2)C1 91607,CCCC(CCCNC(c1ccc(CC)[nH]1)=O)NC(c1sc(C)nc1CC)=O 91608,Cc1ccc2[nH]c(=NCC3CCCC3NC(C3CCCC4(C3)CC4(F)F)=O)sc2n1 91609,C#CC1CN(C(=O)CCOCC(C)C)CCN1C(=O)Cc1n[nH]c(=NC)s1 91610,N1(c2cc(COC)ncn2)C2CCC1CC(CC(C)NC(c1nocc1C)=O)C2 91611,CCCC(C(=O)NC1CCCC(NC(c2ccc(N)c(SC)c2)=O)C1)S(N)(=O)=O 91612,C=C=CC(C)C(=O)NC(c1ccc(F)cc1)CNC(c1ccn(C2CCC2)n1)=O 91613,C1(NC(C(C2CCCCCC2)C)=O)C2CC1N(C(=O)COCCF)C2 91614,CCCCCCC(F)C(=O)N1CCC(CN(C(=O)CC2(O)CCOC2)C)CC1 91615,N1(C(C2CCN(C(C3(N(C)C)CCCC3)=O)C2)=O)CC2CCOC(=O)C2C1 91616,c1(N2C(=O)CC(C(=O)NCCNC(c3ncn(CC)n3)=O)C2)ccc(C#N)cc1 91617,c1(CC(=O)NCC(CNC(CCC(C)N(C)C)=O)O)cc(Cl)cc(Br)c1 91618,c1(CCOC)ccc(Br)cc1NC(=O)C=Cc1nnn(C)n1 91619,CCC(C)CCC(=O)NC(CCOCCO)C(=O)N1CC(N2CC(F)C2)C1 91620,C12(CNC(Cc3cccc(C)c3)=O)CCC(C1)N(C(C1CCCCCCC1)=O)C2 91621,Cc1nnc2ccc(C(=O)NC3CCCC(NC(C4CC(F)C(=O)N4)=O)C3)cn12 91622,C(=O)(CC1C(=O)Nc2ccccc21)NC1CCN(C(c2ncn(C)n2)=O)C1(C)C 91623,Cc1ccc(C(C)NC(=O)CN(C(=O)CCN2CCCCC2)C2CCC2)nc1 91624,c1(NCC=C)[nH]c(=NCC2C(F)(F)C23CCC3)nc2c1ncn2C 91625,CS(=O)(=O)CCC(=O)NCC1CC(NC(c2cn3ccnc3s2)=O)CCO1 91626,N1(C(CC2CC(C)C2)=O)CCc2nc(CNC(=O)C(C)(C)C(C)(C)C)sc2C1 91627,N(C(=NCCN1CCOC(C2CCC2)C1)NC1CCC1)CC1(C#N)CCCC1 91628,C12(C(N3CCC(CNC(=O)C=Cc4cccc(O)c4)C3)=O)CCCN(CCC1)C2 91629,C(=O)(CCC(C)(C)C#N)NCC1CC(NC(c2ccc(SC)o2)=O)C1(C)C 91630,N1(C(c2c(COC)cco2)=O)CCCC2(CCCN2C(=O)Cc2ccon2)C1 91631,C(=O)(CCCCCc1ccccc1)N1CC(NC(C(CC)=CC)=O)C(OC)C1 91632,N1(C(C=Cc2nc(C)c(C)[nH]2)=O)CCCC12CCN(C(=O)C=C1CCOCC1)C2 91633,N1(C(CN2C(=O)CC(C)(C)O2)=O)C(C(=O)NCCN2CCCC2)C2CC(O)C1C2 91634,C(=O)(C1=CC2CCCCCCC12)NC1C(C)(C)CN(C(=O)C=CC2CCCO2)C1 91635,N1(C(COC2(C#C)COC2)=O)CCN(C(=O)C(C)CC=C)C2COCC12 91636,c1(C(=O)NC(CC)CNC(c2ncn(C)c2C)=O)cnc2ncnn2c1C 91637,c1(CCCC(=O)NCCN(C(C2(F)CCOCC2)=O)CC)ccccc1F 91638,C1(C(N2C3CN(C(C4CSCC(=O)N4)=O)CC2C3)=O)CCCC2(CCC2)O1 91639,c1(CC)c(C(=O)NCCN(C)C(C2CCCN2C2CC2)=O)cnc2ncnn12 91640,C(CC(C)C(=O)NC1CCCC1NC(c1cc(C(F)(F)F)n(C(F)F)n1)=O)=CC 91641,c1(C(N(CCCNC(=O)C(C(C)O)N(C)C)CC)=O)ccc(S(=O)(=O)CF)nc1 91642,Cc1nc(C=CC(=O)NCC(C)CNC(=O)C=Cc2nnn(C)n2)cs1 91643,Cc1cnn(C(C)C(=O)NCC2CC(F)(CNC(c3cnn(CCO)c3)=O)C2)c1 91644,N1(C(C2C(C#N)C2)=O)CCC(NC(=O)C(c2ccccc2)N2CCCC2)CC1 91645,C1(CNC(c2c(OC)c(Cl)sc2)=O)CN(C(=O)CC2CC3(CC3)CO2)CC12CC2 91646,c1(OC)c(O)cc(C(=O)NCC2CC(F)CN2C(=O)C(C)OC)cc1C#N 91647,c1(N2CC(C(=O)Nc3nc(C(F)(F)F)cs3)SCC2)ccn2ncc(I)c2n1 91648,CCC(CC)(CCNC(=O)C(C)(CC)OC)NC(=O)CSC(F)(F)F 91649,C(=O)(C(C)(C)ONC(=O)CN(c1ccccc1)C(=O)CN(C)C)OC 91650,C(=O)(C(F)C(C)(C)O)N(C1CCN(C(CC2(C(=C)F)CCC2)=O)CC1)CC 91651,C1(C)(CC)CCC(N=c2[nH]c(=NCc3cncs3)[nH]c3c2CCCCCC3)CC1 91652,N1(C(c2c(OCC)cccn2)=O)CCN(C(C23CC(C)(C2)OC3C)=O)CC1CC 91653,CC1CN(C(C2(C)CCCN2C(=O)Cc2cncnc2)=O)CC1N=[N+]=[N-] 91654,C1(NC(c2c(OC)cccc2)=O)CCN(C(c2ccc(CO)s2)=O)C(C2CC2)C1 91655,Cc1nn(CC(=O)NCC2(O)CN(C(=O)CSCc3ncc[nH]3)C2)c(=O)n1C 91656,C1(c2nnnn2C)(N(CCC(C)C)CCC#N)CC(C)(C#N)C1 91657,C1(C(N2CC(OCC(=O)N(C(C)C)CCl)C2)=O)CCC(NC(C)(C)C)CO1 91658,N1(C(c2cccc(S(C)(=O)=O)c2)C(=O)NC)CCCC2(CC1)CNC(=O)C2 91659,N1(C(CCC#CC)=O)CCN(C(=O)COc2cccc(C)c2)C(C2CCCC2)C1 91660,Cn1nc(C(Cc2ccccc2)NC(N)=O)cc1NC(=O)NC1CC2CC1CO2 91661,C(=O)(CCC[N+](=O)[O-])NC1(C)CCN(C(C2CCCCC2O)=O)C1 91662,c1(C(N2CCCC(CNC(CCCN(C)C)=O)CC2)=O)cnn2c1OCCC2 91663,c1(C(N2CCC(C(C)C(=O)Nc3cn(C)nc3C#N)C2)=O)ncc2ccccn12 91664,c1(N2C(CNC(CC(C)C3CC3)=O)CCCC2)ncnc2sccc12 91665,N1(C(C(C(C)C)N(C)C)=O)CCC2(CCN(C(C3CCCC3O)=O)C2)C1 91666,c1(NC(c2ncn(C)n2)C)ccc(S(=O)(=O)NCC2CSCCO2)cc1Cl 91667,C(=O)(C1=CCCSC1)NC(C(=O)NCc1c(CC)cccc1)C1CCCC1 91668,c1(C(N2CCN(c3nc(C)c(F)cn3)C(CC#N)C2)=O)cc(F)c(C)c(Br)c1 91669,c1(C(=O)NC2C3(CN(C(CC(=O)NCC)=O)C3)CC2)cccc2c1OC(F)(F)O2 91670,CC1CCN(C(=O)CCc2cn(C)nn2)C(CNC(c2cnc(C#N)s2)=O)C1 91671,N1(C(C=CCOC)=O)CCC(NC(c2ncnc(OC)c2F)=O)CC1C1CC1 91672,C(=O)(C(C)(C)C(C)NC(=O)Cc1sccc1C)NCCCCCOC 91673,c1(C(N2CC(N(C(C3(C)N(C(C)=O)CCC3)=O)C)C2)=O)ccc(P(C)(C)=O)cc1 91674,C1(C(=O)NCc2cnc(C)[nH]2)C2CC3C(C2NC(=O)CC2CNC(=O)O2)C13 91675,C=CC(C)(O)CC(=O)NC1(COC)CCN(C(=O)Cc2ccc(C(F)F)cc2)C1 91676,c1(-n2cc(NS(CC)(=O)=O)nn2)ccc(OCCN(C)C)cc1 91677,c1(C(=O)NCC(CNC(c2cc(CN(C)C)on2)=O)OC)nccnc1N 91678,c1(SCC)ccc2cn(CN(C(=O)Cn3ncccc3=O)CC)nc2c1 91679,CC(C)(C)C1=NOC(C(N2CC(C)(C)OCC2CNC(=O)C2=CCCCC2)=O)C1 91680,CCCCC(C(=O)N1CC2CC2(C(=O)OC)C1)NC(=O)CCCCCF 91681,N1(C(CCCCOC)=O)CC(F)(F)CC1C(N1CCN(CCF)CC1)=O 91682,C(CC(O)CC(=O)N1CCCC(NC(C2(C)CCOCC2)=O)C1)SC 91683,C1(C)(C(N2CC(CNC(CNC(CC)=O)=O)C2)=O)CCOC(C)C1 91684,C1(CNC(c2c(SCC)cccc2)=O)CCCCN(C(C2CC2(C)C)=O)C1 91685,C1(O)(CN(C(=O)C#CC(C)(C)O)C)CCCN(C(=O)CC2COCCN2C)CC1 91686,c1(C(N2CC=CC(NC(C(C)(CO)OC)=O)C2)=O)cccc(C)c1C#N 91687,C1(CC(=O)N(CC(CNC(CSCC(C)C)=O)C)C)CCC(=O)C1 91688,C1(CNC(COC(CC)C)=O)CCN1C(=O)CCC1CC1(C)C 91689,C1(NC(C(CC)(F)F)=O)CN(C(=O)CCSC2CCCC2)CCC1O 91690,C(=O)(C1=NOC(C2(O)COC2)C1)N1C(C2CCN(C(CCC=CC)=O)C2)CCC1 91691,c1(C(=O)NC(C(C)NC(CCOC)=O)CO)cc(C)c(OC)c(Cl)c1 91692,N1(C(c2c(CCC)[nH]cc2)=O)CC(CNC(=O)C(C)(C)N(C)C)CC(C)(C)C1 91693,c1(N2CCC(N3C(C)(C(=O)NC)CCC3)CC2)nc(C(C)C)nc(C)c1Br 91694,C1(NC(C=C(C)C(F)F)=O)CC1C1CCCN(C(c2ccc3nc[nH]c3c2)=O)C1 91695,c1(N2C(CN3CCN(C)CC3)CCC2)nc(=NC2CC2F)[nH]c2cccc(F)c12 91696,C1(NC(C(C)NC(C2CCC2)=O)=O)C2CC1N(C(=O)CCN1C(=O)CCC1=O)C2 91697,C1(C(=O)NCCCCN(C(=O)Cc2cc(Cl)ccc2O)C)CC(C2CC2)=NO1 91698,N1(C(C)C)CCN(C(=NCc2nnnn2C)NCc2ccc(F)cc2F)CC1=O 91699,N1(C(C(CC)C(F)(F)F)=O)Cc2n[nH]cc2C1C(=O)N(CCC)OC 91700,N1(C(C=C(CCC)C)=O)CC(CNC(=O)C(C)CC)C(C)(C)C1 91701,N1(C(C2C(C)OC(=O)N2)=O)CC(NC(=O)CCc2ccccc2Cl)CC(C)C1 91702,CCC(O)CC(=O)NCC(C)C(=O)NCCc1ncccc1C 91703,c1(C(=O)NC2C(NC(C(CC)(C)OC)=O)CCCC2)cnc2[nH]cncc1-2 91704,C(C(CNC(C1CCC12CCC2)=O)C(F)(F)F)NC(CC1C(=O)NC(=N)S1)=O 91705,C(=O)(CCCC(=O)OC(C)(C)C)NCCNC(N(C)C)=O.C12CC(F)(C1)C(=O)N2 91706,c1(OC(C)C)ccc(C(N2CC(NC(=O)CC3CCC(O)C3)C2)=O)cn1 91707,c1(C(=O)NC2CCCC(CNC(=O)Cc3csnn3)C2)cc2cc(F)ccc2[nH]1 91708,Cc1cc(C(=O)NC2CC(CNC(C3(CO)COC3)=O)C2)c(C)c(C)c1 91709,C12(C(=O)NCC(C)(C)NC(c3c(C)c(O)ccc3)=O)CCCN1CC(O)C2 91710,N1(C(CCC2(NC(C(CC)C(=O)OC)=O)CCCC2)=O)CCC(F)(F)C(C)C1 91711,c1(ONC(CC2C(C)(C)C(=O)C2)=O)c(C#N)cnn1C1CCCCC1 91712,N1(Cc2c(OC)cccc2Br)CCOC2(CCS(=O)(=O)C2)C1 91713,Cc1cc(C(=O)NCC2CCCN(C(C3CCC3(C)C)=O)C2)cc(O)c1 91714,c1(C(N2CC(CCCCNC(COC(C)C)=O)C2)=O)ccc2ncnc(O)c2c1 91715,Cc1cc(=O)c(C(=O)NC2(C3CCCN3C(C3CCCC34CCC4)=O)CC2)c[nH]1 91716,N1(C(C(C(C)O)C)=O)CCC(C2(O)CN(C(C3CCC4(CCC4)CC3)=O)C2)CC1 91717,C1(NC(C(C)=C(CC)C)=O)CN(C(=O)CCCC(=O)OC(C)(C)C)CC(C)(C)C1 91718,N1(C(CCC(C)C)=O)CCCC2CN(Cc3cc(Cl)ccc3F)CCC12 91719,c1(C(C)=O)ccccc1C(N1CCCC(CNC(C2CC(F)C(=O)N2)=O)C1)=O 91720,c1(C(=O)NC(C(C)(C)NC(C2C(COC)C2)=O)C)[nH]c2ccc(OC)cc2c1C 91721,N1(C(=O)NC(CCCC=C)C(=O)NC)CCc2c(cnn2C)C1C(=O)OC 91722,C1(C(C)(C)C)CCCN(Cc2cc(C3(N)CCC3)cs2)CC1 91723,C1(CNC(Cc2cc(C)ns2)=O)CCN(C(=O)CC2CS(=O)(=O)C2)C1(C)C 91724,c1(C(N(C2CN(C(C(C)OC)=O)CC23CC3)C)=O)cc2sc(C)cc2[nH]1 91725,C(=O)(C(F)C(C)(F)F)NC(C(C)C)CCN(C)C(c1ocnc1C1CC1)=O 91726,C(=O)(C1=CC2CCCCCC12)NCCCC(C)NC(c1cc(C(C)C)on1)=O 91727,N1(C(Cc2ccn(C)n2)=O)CCCC(NC(c2cc(-c3ccccn3)no2)=O)C1 91728,c1(OC)cccc2c1C(C(=O)N1CC=C(CNC(=O)COCCF)CC1)CC2=O 91729,C1(CNC(NC(C2CCCO2)C)=NCCc2cnsc2)Cc2ccccc2O1 91730,c1(C(N2CC(N(C(=O)C(F)CC3CCC3)C)C(O)CC2)=O)nccn2ccnc12 91731,N1(C(C2(OCC)CCOCC2)=O)CC2(CC(CNC(C3CC(C)(C)CO3)=O)C2)C1 91732,C(C)(C(C)(C)C(=O)NCCC(O)C(F)(F)F)NC(c1cccc(C)n1)=O 91733,N1(C(C2=NNC(=O)C2)=O)CC2CCCC(NC(C3CCC4CCC(=O)N34)=O)C2C1 91734,Cc1ncnc(C)c1C(=O)NCC1CC(CNC(=O)Cc2ccsn2)CO1 91735,N#Cc1c(F)cc(C(=O)NCc2ccc(CNC(=O)CCC(F)F)cc2)cc1F 91736,C1(COC)CC(CNC(=O)CC2CC(=O)NC2=O)N(C(c2cc(Cl)c[nH]2)=O)C1 91737,N1(C(C(CC(C)C)F)=O)CCN(C(=O)Cc2ncc(F)cc2F)CCC1C 91738,C1(C#N)(OC)CC(C(=O)NCC#CC(=O)NCCC2CC=CCC2)C1 91739,C(=O)(C(F)CCC(C)(C)C)NCC#CC(=O)NCCN1CCCC(C)C1 91740,N1(C(c2c(OCC)scc2)=O)CCN(C(c2cn(C)c(=O)n2C)=O)C2COCC12 91741,N1(C(CN)=O)CCC2(CC1)CC2NC(c1cc2ncccc2[nH]1)=O 91742,CC1(C)CC(CO)CN1C(=O)C1=NOC(CNC(=O)C=CC2CCCCC2)C1 91743,N1(C(CCc2c(C)cccc2)=O)CC2CCCC(CNC(=O)CN3CCC3)C2C1 91744,CC(C)(C)C(=O)N1CCCC1C(=O)NC1(CNC(=O)C=C2CCC2)CC1 91745,C(C(=O)N1CC(CN(C)C(c2ccc(-c3cccnc3)s2)=O)C1)(C(C)C)OCC 91746,c1(CNC(=O)CNC(c2cccnc2)=O)ccc2nonc2c1 91747,c1(C(=O)NCCC2(O)CCCN(C(C=C(C)C(C)C)=O)C2)nc2c(s1)CCCC2 91748,CC1(CNC(=O)NC(CCC(=O)O)c2ccccc2)COc2ccccc2O1 91749,O(NC(=O)C1(N(C(=O)C=CC(C)(C)C)C2CC2)CCC1)CCC=C 91750,O=[N+]([O-])c1cccc2c(NCC(O)CC3CC3)nc(Cl)cc12 91751,C1(O)(CNC(C(c2cccc(OC)c2)C)=O)CCCN(C(C2(SC)CC2)=O)CC1 91752,c1(OC)ccc(S(N)(=O)=O)cc1NC(C1CSCCN1C(c1csc(Br)c1)=O)=O 91753,C=CC(C)(CCOC)C(=O)NCC1=CCN(C(=O)CCC2CCN(C)CC2)CC1 91754,N1(C(C2C(=C)C2)=O)CCC(C2N(C(C3CCN(C)C3=O)=O)CC2(C)C)CC1 91755,c1(C(=O)NCC(C23CCC(CC2)C3)O)ccccc1Br 91756,N1(C(CCOCCC)=O)CCn2nc(CNC(C3CCCOC3)=O)cc2C1 91757,N1(C(C2C(C(C)C)C2)=O)CCCN(C(c2ccc(CCF)cc2)=O)CC1 91758,c1(C(N(CC(C)CNC(=O)COC2CC2)C)=O)ccc(C=C2CCCCC2)cc1 91759,C12(OC)CCC1CN(C(c1cn(C(C)(C)C)nn1)C(=O)NCCCSC)C2 91760,c1(OC)cc(OC)c(CN2CCN(C(c3ccnc(F)c3F)=O)C3CC23)c(Br)c1 91761,CC1(C)C(NC(c2cncnc2)=O)C(C)(C)C1NC(c1ccc(F)s1)=O 91762,C#CC1(C(=O)Nc2cnccc2CO)CN(C(c2cc(C)on2)=O)C1 91763,c1(CC)cc(N)ccc1C(=O)N(C1CCCCC1N(C(=O)C(N)=O)C)C 91764,N1(C(C(C)C)=O)CCC(CC(C)NC(C2CCCN2C)=O)CC1 91765,N1(C(C=CC(=O)N(C)C)=O)CCCC1C(=O)NCCc1ccncn1 91766,C1(NC(CC2C(C)(C)N(C(=O)Cn3[nH]cnc3=N)CC2)=O)CCC(C2CC2)CC1 91767,C1(C(=O)Nc2ccc(COC)cc2)CC1C1CN(C(c2ccc(CO)o2)=O)C1 91768,c1(C2(C(=O)O)CC(NC(=O)C(c3ncc(F)cc3Cl)(F)F)C2)ccc(F)c(F)c1 91769,c1(CNCC(c2ccccc2Cl)(C)O)cc(Cl)cc(Cl)c1 91770,c1(C(=O)NCC2OCC(CNC(=O)C=Cc3ccccn3)C2)cc(=O)c(O)c[nH]1 91771,C(C)(CNC(=O)Cn1cc(C(C)O)nn1)(CC(C)C)NC(C(CCOC)OC)=O 91772,Cc1nn(CC(F)F)cc1C(=O)NC(C)CN(C)Cc1cn(C)nn1 91773,C1(C)(CNC(CCC=C)=O)CCN(C(c2ccc3c(c2)CC3)=O)CC1 91774,Cc1cc(O)nc(C)c1C(N1CCN(C(c2oncc2C)=O)CC(C)C1)=O 91775,C=C(CC)CN=c1nc(N(CCCN2CCOCC2)C)c2c([nH]1)CCC(C)C2 91776,CC1CCc2[nH]nc(C(N3CCC(NC(=O)C4=CCSC4)C3C(C)(C)C)=O)c2C1 91777,C1(C(=O)NC(CN(C(c2cccc(F)c2)=O)CC)C)CCOC(=O)CC1 91778,c1(C(C)CNC(=O)N(C2CC2)CC2CCOC2)ccccc1Cl 91779,C1(C(=O)NC(CC)CO)CN(C(=O)C(C)NC(=O)Cc2cccs2)CCC1O 91780,CCS(=O)CC(=O)NC1(C(=O)NCCOCC(F)(F)F)CCSC1 91781,c1(OCC(=O)NCC2C(NC(COCC)=O)C2)cccc(C(N)=O)c1 91782,c1(C(n2nnnc2C2(NC3CS(=O)(=O)C3)CCC2)C)ccc(F)c(Cl)c1Cl 91783,C1(NC(c2c(C(N)=O)nccc2)=O)CCCC(NC(=O)CCCCC2CC2)CC1 91784,C(c1ccccn1)=C(C(N1CCC(N(C(C2CC(C)(O)C2)=O)CC)C1)=O)C 91785,Cc1cnc(C=CC(=O)NCC2CCN(C(=O)CN(C3CCCC3O)C)C2)[nH]1 91786,C12(NC(C(C(C)C)SCC)=O)CCCC(NC(c3ccc(C)cc3N)=O)(C1)C2 91787,C(CC(C)(C)C(=O)NC(CNC(c1ccccc1NC(N)=O)=O)CO)OC 91788,N1(C(C(C(C)NC(C=CC(=O)OC)=O)C)=O)CCCC2CN(C)CC12 91789,C1(N(C(=O)CCC2CC(F)(F)C2)CC)CCCN(C(=O)C(C)CNC(N)=O)C1 91790,N1(C(C2(NC(C)=O)CCC2)=O)CCCC(CNC(=O)Cc2csc(COC)n2)C1 91791,C1(NC(CC=C=C)=O)COC2(CCCN(C(=O)Cc3cc(OC)ccc3Cl)C2)C1 91792,N1(C(c2nc(CCC)oc2)=O)CCC2(CCCC2NC(c2c[nH]c(=NC)o2)=O)C1 91793,N(C(=NCCC(C)CC(C)(C)C)NCCc1nn(C)cc1C)C(C=C)C 91794,N1(CC)CCN(C(C2CCN(C(=O)CC(C)(C)C3CC3)CC2C)=O)CC1(C)C 91795,C1(C)(NC(C(C)c2ccco2)=O)CCN(C(=O)C(O)C(F)(F)F)CC1 91796,c1(C(=O)NCC23OCCC(NC(C(C(C)C)C)=O)(C2)C3)nnn2c1CCCCC2 91797,c1(OC)ccc(Br)c(F)c1CN1CCOC(C)CC1 91798,c1(-c2nc(-c3ccc(-c4ccc(C)cc4)s3)on2)ccc2ncccc2c1 91799,C1(C(C)C(=O)NCC=CCl)CCN(C(=O)C(C)(C)N2CCCC2)C1 91800,C(C)(CO)(C(=O)NCC1(F)CC(NC(c2cc(Cl)n(C)n2)=O)C1)NC(C)=O 91801,CC1CN(C(=O)CC2(O)CCC2)CC(C)C1NC(c1cc(F)n(C)n1)=O 91802,Cc1cc(Cl)cc2[nH]c(C(=O)N(CC(O)CNC(C3CS(=O)(=O)C3)=O)C)cc12 91803,C(=O)(C1=CCCOCC1)N1CC(C)CC(NC(c2c(CCC)occ2)=O)C1 91804,N1(C(C(C2CC2)OC)=O)CC(C)(OCC(=O)N(CCCF)C)C1 91805,CC(C)C(C)CC(=O)NC1(CNC(C2CC3CCCC23)=O)CCOCC1 91806,N1(C(C(CC(=O)OC)C)=O)CC(NC(c2c[nH]c(C)c(Cl)c2=O)=O)C2(CCC2)C1 91807,N1(C(C(=O)NCC)=O)CCC2(CC(NC(=O)C(C(C)(C)C)n3ccnn3)C2)C1 91808,C=CC(C)(O)CC(=O)N1CCC(c2cn(CCNC(=O)C(C)(F)F)nc2)CC1 91809,C1(NC(c2ccc(N(CCC)CC)cc2)=O)CCN(C(c2nncs2)=O)C1(C)C 91810,c1(COC)ccc(NC(=O)C(CC2C=CCC2)N2CCC(CN3CCCC3)C2)s1 91811,N1(CC(CC)CC)CCC(C2CCN(C(c3ccc(C)o3)=O)CC2)C1 91812,C=CCCCCCCC(=O)NCC(=C)CCNC(C1CCCCC12CCC2)=O 91813,c1(Cn2cc(C3CCN(C(c4ccc(C(C)=O)s4)=O)C3)nn2)ccc(Cl)nc1 91814,c1(NC(C(C(C)NC(=O)C(C)(Cl)Cl)C)=O)cc(O)cc(F)c1 91815,N1(C(Cc2cc(OC)no2)=O)CCCC2(CCCN2C(c2cc(O)ncn2)=O)C1 91816,c1(CCC)ccc(S(=O)(=O)N2CC3CCC(C2)N(C(c2nnc(C)o2)=O)C3)cc1 91817,c1(C(=O)NCCN(C2CCCC2)C(C=Cc2ncc(C)[nH]2)=O)ccc(Cl)cc1O 91818,c1(C(=O)NC(CNc2nccc(OCCOC)n2)C)ccc(C)c(C)c1O 91819,C(=O)(C1CCCc2scnc21)N1CCC(N(C(C2C=CCCC2)=O)CC)CC1 91820,c1(C(C(=O)N(CCCN(C(=O)CSCc2cccnc2)C)C)=O)ccc(Cl)s1 91821,C1(C(=O)NCCCCNC(C(CC)n2cncn2)=O)CCC2(CCOCC2)CO1 91822,C1(NC(COC(CC)CC)=O)CN(C(=O)C(CC)C(C)C)CC12CC2 91823,c1(CNC(c2cc(C)on2)=O)ccnc(C(N2CCC(C(C)O)C2)=O)c1 91824,C(c1cccc(O)c1)=CC(=O)NC1C(OC)CN(C(=O)C=Cc2ccnn2C)C1 91825,Cn1nc2c(c1C(=O)NCc1c(F)ccc(CO)c1F)CN(c1ncccn1)CC2 91826,S(=O)(=O)(c1ccccn1)N1CC(NC(C2N(C)CCC2)=O)(CO)C1 91827,N1(C(c2cccc(-c3ccccc3)c2)=O)CC2CCC2(C(C2CCN(C)C2)=O)C1 91828,Nc1cc(C(=O)NCc2cc(O)nc(CNC(=O)C=CCO)n2)cc(O)c1Cl 91829,C1(C(=O)NCC(C)(CO)NC(c2cc(F)n[nH]2)=O)CC2CCCC(C1)C2 91830,C(=O)(C1=CC2(CCOC2)C1)NCC1(OC)CN(C(C2(C)CC3CCC2C3)=O)C1 91831,CC1(C)CCCC(C(=O)NCC23CC(NC(C4CCS(=O)(=O)C4)=O)(C2)C3)O1 91832,C1(NC(c2c[nH]cc2C2CC2)=O)CCCCCC1NC(C1CCSCC1)=O 91833,c1(CC(N2CC(n3cc(-n4nc(C)c(Cl)c4)nn3)C(C)C2)=O)cccc(Cl)c1C 91834,C=C(Br)CC(C)(C)C(=O)NCCC1CCC(NC(c2cnnn2CC)=O)C1 91835,CC(C)(O)C(C)(C)CNC(C1C=CC(NC(=O)CCc2cccnc2)C1)=O 91836,N1(C(CC(C)=C(C)C)=O)CCC2(CC1)CC(CNC(c1ncn(C)n1)=O)C2 91837,C1(OC)(CNC(=NCc2cc(C)on2)NC2CN(C(C)C)CC2C)CCSCC1 91838,C(=O)(CCCCC(C)CC)NCC(CCC)C(=O)NCc1nn(C)c(=O)n1C 91839,c1(C(=O)NCCOC)ccc(N(C2CCCCC2NC(=O)C(=O)NC)C)cc1 91840,CCCCC(O)C(=O)N1CCC(CNc2ncc(C)c(O)n2)C1 91841,c1(CCC(=O)NCCN(C(c2cc(O)nc(C)n2)=O)CC)csc2ccccc12 91842,C1(CNC(c2nc(COC)sc2)=O)C2CCC(C2)N1C(=O)CC1C=CCCC1 91843,C(C)(C)(CC(F)C(=O)NCCC1CCOCC1)NC(C(NOC)=O)=O 91844,c1(C(=O)NCC(C)N(C(c2cccc[n+]2[O-])=O)CC)cnc2c(cnn2C)c1N 91845,N1(C(Cc2n(C)ncc2)=O)CC2CC2C1CNC(C1(c2ccsc2)CC1)=O 91846,Cc1nc2ncc(C(=O)NC3CC(NC(C4(C)CSC4)=O)C3)c(=O)n2[nH]1 91847,N1(C(c2c(C)n[nH]c2)=O)CCc2nc(O)cc(C(N3CCCC(F)CC3)=O)c2C1 91848,C1(CNC(C2(CN)CCCC2)=O)CCCC2(CCC2)O1 91849,c1(CCC(=O)NCCC2CN(C(C3CC4CCC4C3)=O)CCO2)cccc(O)c1 91850,C(CC(C(=O)NC1C=C(C)CCC1)NC(=O)Cn1cccc1)=CC 91851,c1(C(N2CC(C)(NC(c3cn(CC(CC)O)nn3)=O)C2)=O)ccc([N+](=O)[O-])[nH]1 91852,C=CCC(C)C(=O)N=S(C)(=O)c1cnn2c1CN(C(=O)C(C)C(=O)OC)CC2 91853,CC1(C(=O)NCC(O)C(F)(F)F)CCCN(Cc2cc(Cl)ccc2O)C1 91854,C12(C(=O)NC(c3ccccc3)CNC(C3(CF)CCC3)=O)CCN(CC1)C2 91855,C=CCCC(F)(F)C(=O)N1CCCOC(CNC(c2c(C)noc2CCC)=O)C1 91856,CC1(C)C(C(=O)NC(C2CCCCC2)C(N2CCC(F)(F)C2)=O)C1(F)F 91857,S(=O)(=O)(c1ccc(Br)cc1NCc1ccc(C2CC2)cn1)NC(CCC)CO 91858,N1(C(C(=Cc2ccco2)C)=O)CC2CCOC2(CNC(c2cncc(C)n2)=O)C1 91859,N1(C(C2C(CCOC)C2)=O)CCOCC(NC(=O)C(F)(F)CN(C)C)C1 91860,Cc1ccc(F)c(CNC(C2CCC(CNC(C3CC4CCC4C3)=O)O2)=O)c1 91861,c1(CC)ccc(C(=O)NCC2(C)CC(NC(=O)C(C)(C)n3cccn3)C2)nc1 91862,CCCC(CCC)C(=O)NC1CC(O)CN(C(=O)C(C2CCOCC2)F)C1 91863,N1(C(c2n(C)nnc2)=O)CCC2(NC(c3ccncc3Br)=O)CCCC12 91864,C(=O)(C(CC(F)F)c1ccccc1)N(CCCNC(C(C=C)(C)O)=O)CC 91865,N1(C(c2c(CCC)nco2)=O)CCC(C)(C)C1C(=O)NCc1nccn1CCC 91866,CC(C)CCC(O)C(=O)NC(C)(C)CC=CC(=O)NC1CCN(C(C)C)C1=O 91867,C1(C(N2CC(O)(C(C)(C)CNC(c3sccc3CO)=O)C2)=O)CC(=O)CCO1 91868,C1(NC(Cc2nc(CC)sc2)=O)CC2CCC(C1)N2C(=O)CC1C(=O)ON=C1C 91869,N1(C(C2CC(CNC(=O)CSCC(F)F)C2)=O)CCOCC2(CC2)C1 91870,c1(C(N2CCC(O)(C(=O)OC)CC2)C(=O)NCCOCC)nc(Br)c(C)cc1Cl 91871,C#CCCN=C(NCC(C)Cc1cccs1)NC1CC(CNC(=O)OC(C)(C)C)C1 91872,C1(C(N(C(C)C)CCNC(C2CCN(CC(F)(F)F)C2)=O)=O)CCCOCC1 91873,Cc1cc2cc(C)c1NC(=O)C(=O)N2.N1(CC(C)O)CCCCC1C1CC1 91874,c1(CC(C)C)ccc(C#N)c(NC(C)CNC(=O)Cc2cc3ccccc3s2)n1 91875,CCN=c1[nH]c(C)c(C(N2CCCCC2CNC(C2CCNC2=O)=O)=O)s1 91876,c1(C(N2CC(C)N(C(c3cnn4ccsc34)=O)CC2)=O)cccc2ccsc12 91877,CC1CC(CNC(=O)C(F)(F)C2(O)CCC2)CN1C(=O)COc1ccccc1Cl 91878,Cc1cc(=NC(C)CC2CCOC2)[nH]c(=NCc2nnc3n2CCOC3)[nH]1 91879,Cc1ccc(C)c(CC(=O)NCCCC(C)NC(c2ccn(C(F)(F)F)n2)=O)c1 91880,C1(C(N2CCC(N(C(CN(C(C)=O)C)=O)C)C2)=O)COCCN1C 91881,N1(C(CCC)=O)CCC(NC(c2cc(CC)nnc2C)=O)CC1C 91882,C=CC(CCC)CC(=O)N1CCOC(CCCNC(=O)CCN(C)CC)C1 91883,n1(CC)cc(Br)c(C(N2CC(NC(=O)C=Cc3cncn3C)C3CC23)=O)n1 91884,c1(C(N2CC(O)(CNC(CSCC#C)=O)C2)=O)nc(C)[nH]c2nccc1-2 91885,N1(C(Cn2ccc(C)n2)=O)CC2CN(C(c3ccc4nsnc4c3)=O)CC2C1 91886,c1(C(=O)NCCCNC(C2CC(O)C(F)C2)=O)cncc2c1CCCC2 91887,c1(C(=O)NCCC(CCNC(C)=O)C)c[nH]cc(Br)c1=N 91888,N1(C(c2nc(C(OC)OC)sc2)C(=O)NC(C)CC)CC(N(C)C)C(C(N)=O)C1 91889,C(CCC(C)(C)NC(=O)C(COC(C)C)N(C(C)COC)C)OC 91890,Cc1cccc(S(=O)(=O)CCCN2CCn3c(C(F)F)nnc3C2)c1 91891,C(=O)(C1CC=Cc2ccccc21)NCC(C)(CO)NC(=O)Cn1cccc1 91892,N1(C(C(C=CC)O)=O)CCCCC(N(C(=O)CN(c2ccc(Cl)cc2)C)C)C1 91893,C(=O)(C1=CCCCC1C)N1CC(O)(CN(C(CCCOC)=O)C)C1 91894,C1(N(C(C(C)OCC)=O)CC)CCCN(C(c2n[nH]c(=N)s2)=O)C1 91895,C1(CNC(C(CC)SC)=O)CCCN(C(=O)CSc2ncccn2)CC1 91896,N1(C(=O)Nc2c(C(=O)NC)n(C)nc2)CCC2NC(=O)NCC2C1 91897,N1(C(CC)=O)C2CCC1C(CNC(=O)C=Cc1ccc(-c3ccc(Cl)cc3)s1)C2 91898,C1(CNC(COCCC)=O)CC2COCC2N1C(c1c(F)ccnc1F)=O 91899,c1(C(N2CC3CC2CC3O)C(=O)NCCCC)ccc(C)c(Cl)c1 91900,C(=O)(C(O)C1=CCCCC1)NC1(c2cn(C3CC(C(=O)O)OCC3)nn2)CC1 91901,C1(NC(c2c(C)ncn2O)=O)CN(C(C2OCC3COCCC23)=O)CC1N=[N+]=[N-] 91902,N1(C(C(C(CC)O)C)=O)CC=C(CCNC(c2ccnn2CC2CC2)=O)CC1 91903,CC1(C)CCN(C(=O)CC2CCC(=O)NC2)C1C(=O)NC1(CF)CCC1 91904,CC(O)(CC(=O)NC1CCCC1C(=O)NCc1cc(F)c(Cl)cc1Cl)CC(=O)O 91905,C(=O)(CC(C(C)CC)NC(C1(CC)CCOC1)=O)NC(C=C)C 91906,C1(NC(c2c(N(C)C)ccnc2)=O)CCN(C(=O)CC2(C)CCC2)CC(O)C1 91907,CCC(C(O)C(F)(F)F)N=c1cccc(S(=O)(=O)NCC2(C)CC3(CC3)C2)[nH]1 91908,c1(C(C(=O)Nc2cccc(OC3CC3)c2)O)cc(F)c(F)c(F)c1 91909,C1(OC)(OC)CCC1C(=O)NC1CCCC1CNC(=O)C(c1ccccc1)OC 91910,c1cc2[nH]c(=NCCCOc3ccncc3)[nH]c(=NCC3CCCS3)c2s1 91911,CN(CC(=O)NC1CCCCC1)N1CCC(OCCO)CC1 91912,C12COCCN(C1)C2=O.C1(OC2(CNC(CC3CC(C)C3)=O)CC2)CCOCC1 91913,CC(C)(C)CC(O)CC(=O)N1CC=CC(C(=O)NCC(c2ccccc2)F)C1 91914,C1(O)(C(N(CC(C)NC(c2ccc(C(=O)CF)cc2)=O)C)=O)CC(C)(C)C1 91915,CCC(C)(CC)C(=O)NCCC(CNC(c1[nH]ccc1C)=O)OC 91916,CCCC(O)C(CO)NC(c1cnn(CCNC(=O)CSCCC(C)C)c1)=O.C(C)=O 91917,c1(CC(=O)NCCC2CCN(C(C(CSC)OC)=O)C2)ccc(C(C)(C)C)cc1 91918,N1(CC(N2C(CNC(Cc3cc(C)ns3)=O)C=CC2)=O)CCNC(=O)C1 91919,Cc1ccc(C#N)c(NC(C2C3CC2N(S(=O)(=O)c2ccncc2)C3)=O)c1 91920,c1(CN(C)Cc2cc(F)ccc2-c2ccc(N)cn2)n[nH]c2c1COCC2 91921,Cc1c(F)cccc1S(=O)(=O)N1CC(O)CC1C(=O)NC(C)CCO 91922,N1(C(COC2CCCC(C)C2)=O)CCN(C(=O)Cc2ccc(F)nc2)CCC1C 91923,n1(CCC(N2C3C(NC(C(C)(C)F)=O)CC(C3)C2)=O)ccc2ccccc12 91924,c1(Nc2ccc(NCc3ccc(C)n(C)c3=O)cc2)sc2ccccc2c1C#N 91925,C1(NC(c2cnc(SC)s2)=O)CN(C(c2cc(C)nc(Cl)c2)=O)CCC1C 91926,c1(C(C(=O)NCC(C(C)C)NC(C2(CO)CCOCC2)=O)C)c(Cl)cccc1Cl 91927,C=CC(C)(CC)C(=O)N1CCN(CC(N2CCCN(C(C)=O)CC2)=O)CC1 91928,c1(C(=O)NC2CCN(C(CN(C(C)=O)C)=O)C2(C)C)nn(C)c2c1CCC2 91929,C(=O)(C(O)CC(C)(C)C)NC1C2CC(NC(c3c(OC)ccs3)=O)CC21 91930,N1(C(c2c(C)[nH]c(=N)s2)=O)CCCN(C(C2CC23CCCCC3)=O)CC1 91931,c1(CN2CCC(NS(CCC)(=O)=O)C2)ccc(OC)c(F)c1 91932,N1(C(CC=C)=O)CC(CNC(=O)C(C2CC2)SC)CC12CCC2 91933,c1(NCCOC)cc(C(=O)NC2CCCC2CNC(c2nc(C)no2)=O)ccn1 91934,C1(C(N(C2(C(N(CC(CC)C)C)=O)CCC2)C2CC2)=O)C2CCC(F)C12 91935,C#CC1CN(C(=O)C(CNC(C2CC(=C3CCC3)C2)=O)C(C)(C)C)CCN1C 91936,C1(OCC)CC2(C1)CC2C(N1CCC(C(C)NC(c2nocc2C2CC2)=O)C1)=O 91937,C(=O)(C(CC)CCCC)N(C(C1CC=CCC1)C(=O)Nc1cccc(CC)c1)CC 91938,C12(CNC(c3c(C)coc3)=O)CCC(CC1)N2C(c1cc2scnc2[nH]1)=O 91939,C=Cn1cc(C(c2nnnn2Cc2ccccc2OCC)NC2CC2CF)cn1 91940,C1(OC)CC2CC1CN(C(=O)CC1(N(C)C(c3cnncc3C)=O)CC1)C2 91941,c1(C(=O)NCCCOCCN(C(CC2CCC(C)O2)=O)C)cccc(Cl)c1 91942,C(C(=O)N=c1c(Cl)c[nH]cc1I)Oc1c(OCC)cccc1 91943,c1(NC(CCOC)C(C)C)[nH]c(=NC(C)c2cncc(Cl)c2)nc2scnc12 91944,c1(CC(=O)NCC(C)N(C)C(C2CN3CCC2CC3)=O)ccc(Br)cc1F 91945,c1(C(N(CCNC(C2CCCCC2F)=O)C2CC2)=O)ccccc1F 91946,C1(NC(C2C(C)C2)=O)CN(Cc2cc(Cl)cc(Cl)n2)CC1C#N 91947,C(=O)(C(C)(C)C(=O)N1CC(NC(C2C3CNC(=O)C23)=O)C(F)C1)OCC 91948,c1(C(=O)NCC(CC=C)NC(=O)C(C)(C2CC2)OC)n[nH]c(C)c1[N+](=O)[O-] 91949,Cc1cc(O)ncc1C(=O)NC1CC1CNC(c1ccc(O)c(Cl)n1)=O 91950,C1(C(c2nnnn2CCC2CC2)NC2C(CCC)C2)CC12CCCCC2 91951,N1(C(C23N(C(c4c(C)cn(C)n4)=O)CCC2C3)=O)C2CCC1CC1(C2)N=N1 91952,N1(C(CC(=C)C)=O)CCC2(C1)CN(C(c1ccnn1C(F)F)=O)C2 91953,Cc1nsc2ncc(C(N3CCCC4(C3)CN(C(C3CCCOC3)=O)C4)=O)cc12 91954,c1(C(=O)OC)cc(Cl)c(N2CCCC(N(C)C(C3CC=CCC3)=O)CC2)nc1C 91955,CC1CCC(C)(C(=O)NC2CC(NC(c3cncc(N)n3)=O)C2)C1 91956,c1(NC(C2CC(O)CN2Cc2ccc(Br)nc2)=O)c(F)cc(F)cc1[N+](=O)[O-] 91957,c1(-c2cn(C3CC(C)(O)C3)nn2)ccc(N)cc1 91958,c1(C(=O)NCC(C(C)C)NC(c2cc(OC)ncn2)=O)sc2cccnc2c1Cl 91959,C(CC(=O)NC12CC1CN(C(c1ncoc1C1CCC1)=O)C2)(C(C)C)OCC 91960,C(CCCCCNC(=O)CC1CCN1C(=O)C(C1CC1)OC)OC 91961,c1(C(N2C(CC)CN(C(=O)CC3=CCCCC3)CC2)=O)cc2cc(Cl)cnc2[nH]1 91962,c1(CC)ncncc1C(N1CCC(CNC(C23COC(CO)(C2)C3)=O)C1)=O 91963,c1(C(c2nnnn2C(C)C)NCC(CC=C)(C)C)c(F)cnc(Cl)c1C 91964,N1(C(c2cc(C)[nH]c2)=O)CC23CCCC2(C1)CN(C(=O)CCc1ncccn1)C3 91965,CN1CCc2cc(C(=O)N(C3CC(NC(C4CCCC(C#N)C4)=O)C3)C)ccc21 91966,c1(CN2CC(F)(C(=O)NCC)C2)csc2ccccc12 91967,C(N=c1[nH]c2cc(Br)ccc2o1)C1C(C)CN(C(C2CCOC2)=O)C1 91968,c1(OC)ncnc(N2CCC(O)C(C(=O)Nc3c(F)cccc3Cl)C2)c1C 91969,N1(C(c2c(C)cc(Cl)cc2)=O)CCCC(C2CCN(C(=O)C(O)C(C)C)CC2)C1 91970,N1(C(=O)CCCc2ccc(C3CC3)cc2)CC2CCC(C1)N(C(=O)CO)C2 91971,c1(C(N(CC(c2ccccc2)CC)CC)=O)ccc(C(F)(F)F)s1 91972,N1(C(CC(C)SC)=O)CCOCC1CC(=O)NOC1CCC(O)C1 91973,CCC(C(=O)N1CC(C)C(C)(CNC(C2CC(O)C2)=O)C1)C(F)(F)F 91974,CCC(C)C(CN(C)C)CCNC(=O)CC(CNC(=O)C(C)OC)C1CCC1 91975,C1(NC(c2cc(C)[nH]n2)=O)CC(O)CN(C(c2ccc(-c3ccccc3)o2)=O)C1 91976,c1(NCCOCC=C)cc(=NC2CCOc3ccc(F)cc32)[nH]c(COC)n1 91977,C1(CCNC(C(C)C2CC2)=O)CCC(NC(=O)CN2CCOC2=O)C1 91978,c1(C(N2CCC(NC(c3n(CC#C)cnn3)=O)(CO)C2)=O)c(Cl)ccc(F)c1F 91979,c1(OC)c(C(=O)NCC(C)N(C(=O)COC2CCOC2)C)cc(Br)cc1F 91980,CN1CCOCC1CC(=O)NC12CC1CN(C(c1cn(-c3nccs3)nn1)=O)C2 91981,C1(CNC(C2CN(C(C)=O)C2)=O)CC(F)(CCCN(C)C)C1.C1C(=O)N1 91982,c1(C(=O)NC(CCNC(c2cc(C(C)C)no2)=O)(C)C)cc2c(ccn2C)[nH]1 91983,C1(C(N2CCCC(N(C(Cc3c(C)cco3)=O)CCF)C2)=O)CCCCC1(F)F 91984,C1(C(=O)NCC(CC)(C)O)COCCN1C(c1cc(=O)cc[nH]1)=O 91985,C=CCC(C)(C)CC(=O)NCC1CCCN1C(c1cc(C)c(C)nc1O)=O 91986,C1(CNC(CSCCC(C)C)=O)CN(C(=O)CC(C)F)CC2(CCC2)O1 91987,N1(C(=O)CN2CCN(C)CC2)CCN(C(=O)NC)CC1.C12(CC1)C(=O)N2C.CO 91988,CC1=NOC2(C1)CC(C(N1CC(NC(C3CCS(=O)CC3)=O)C(C(F)F)C1)=O)C2 91989,C1(C(=O)NC(C(C)C)C2CCC2)(CC)CCN(C(c2c[nH]nc2C)=O)CC1 91990,N1(C(C(CCC)O)=O)CC2(C1)SCCC2NC(=O)CCc1cncc(OC)c1 91991,c1(CNC(C2CC(CCNc3cc(OC)ncn3)C2)=O)ccc(C)c(Cl)c1F 91992,C1(NC(C2(CC#C)CCCC2)=O)CCC(C)(NC(c2cc(Cl)ncc2O)=O)CC1 91993,Cc1noc(C)c1CCC(=O)NC1(C)CC(NC(C2CC23CC3(F)F)=O)C1 91994,N1(CC(C)NC(=O)OC(C)(C)C)CCC2(CC1)OCCc1ccccc12 91995,c1(NC(CCC)CCCNC(=O)CCC(N)=O)ccc(S(C)(=O)=O)cc1[N+](=O)[O-] 91996,C1(C(=O)NC2C(CNC(C)=O)C2)CCc2ccnn2C1.c1sccc1C(C)(C)C 91997,Cc1ccc2[nH]c(C(N3CC(CCCCNC(=O)C#CC4CC4)C3)=O)cc2c1 91998,n1(CC)cc(Br)cc1C(=O)NC(C1(O)CN(C(C2CC23CCC3)=O)C1)C 91999,C1(C(=O)NC(C)CN(C(=O)CSCC(F)F)C)(OCC#C)CCCCC1 92000,CC(Cc1ccco1)N=c1[nH]c2c(c(=NC(C)c3ccncn3)[nH]1)CCC2 92001,C=CCC(CC=C)C(=O)N1CCCCC1C1CCN(C(C2(CCO)CC2)=O)CC1 92002,O=C1NCC2(CO1)COC(CF)CN2C(C1C2CC=CCC12)C(=O)N1CCCC1 92003,C1(NC(=O)C=Cc2cncs2)CCN(C(C2CCCNC2=O)=O)CC12CCC2 92004,CC(C(F)C(=O)NC1C2CC3CN(C(c4ccc(F)cc4)=O)C1C3C2)C(F)(F)F 92005,C=CCC(C(=O)N1CCC(CC(C)NC(=O)C(=O)NC2CC2)CC1)NC(C)=O 92006,C1(C(=O)NC(CCC)CCO)CN(C(C2(SC)CC2)=O)CCC1(C)C 92007,c1(C(=O)NC(C(=O)N(C(COC)COC)C)C2CCCO2)c[nH]cc1C(C)C 92008,c1(C(N2CCC3CN(C(=O)CCF)C3C2)=O)cc(Cl)cc2c1CCC2 92009,N1(CCC)CCc2nc(C(=O)N(CCO)Cc3ccccc3)cn2CC1 92010,N1(C(C2(CCC)CCC2)=O)CCC2C(C(=O)NCC(F)(CC)CC)C2C1 92011,CCCCCCCC(O)C(F)(F)C(=O)NCCN(C(=O)CC1CCCCCC1)C 92012,c12ccc(cc1Br)S(=O)(=O)NC1(C)CN2CCO1.C(CCCCC1CC1)OC 92013,c1(OC)c(Cl)nc[nH]c1=NCCC1CCNCC1.C(=O)CC1=NN(C)C(=O)C1 92014,c1(C2(F)CC(C(=O)NC(C)CCN(C)C(C3CC3C)=O)C2)cccc(F)c1 92015,Cc1cccc(C(N2CCC(C(N3CCCCC(C)(F)C3)=O)CC2C)=O)c1C#N 92016,N1(CCC)CCC(C(=O)NCCN(C(=O)C(O)Cc2ccc(F)cc2)CC)CC1 92017,C(=O)(C(C)(CNC(=O)C(N)=O)CC)N1CCC(OCC)C1 92018,c1(OC)cccc2cc(C(=O)NC3CCN(C(=O)C(F)=C(C)C)C3)oc12 92019,C1(CN(C(c2cc(C(F)(F)F)ncn2)=O)CCF)CCN(c2ncns2)C12CC2 92020,N1(C(CCN(C(=O)CC2C=CCC2)C)=O)CCCCC1CF 92021,c1(C(=O)NCC(C(C)C)NC(c2ccsc2Br)=O)ccnc(C2CC2)n1 92022,c1(OC)cccc(C)c1NC(C1(CNC(c2ccc(C(F)F)o2)=O)CCCO1)=O 92023,C1(CC(N)=O)(NC(C2CC(=C)C2)=O)CCN(C(C2CC3(CCC3OC)C2)=O)CC1 92024,CC1CN(C(c2cc[nH]n2)=O)CC1NC(c1ccc(-c2ncon2)cc1)=O 92025,c1(C(=O)NC(C(=O)NC2(C)CC(O)(CO)C2)CCF)cccc2occc12 92026,C(=O)(C(=O)CC(C)C)NC(C(=O)NCC(CC)C#N)(C)CO 92027,C12(C(CNC(=O)C(Cl)=CCl)NC(=O)CSCc3ncc[nH]3)CCC(CC1)C2 92028,N1(C(C=CCC)=O)CCCC(CC(=O)NC2CCCSCC2)CC1 92029,C1(CC(=O)NCCOC(C)=O)CCCN(C(=O)Cc2cn(C)nn2)C1 92030,c1(C(N2C(C3CCN(C(C(CCC)O)=O)C3)CCC2)=O)coc2ccc(C)cc12 92031,Cc1cc(NC(C2CC(C)(C)CN2C(c2cccc(C)c2N)=O)=O)cnc1Cl 92032,c1(C(N2CCC(OCCNC(C(C)OCCC=C)=O)CC2)=O)ccc(C)nc1C 92033,c1(C(N2CC(C)CC(NC(C3(OCC)CCCC3)=O)C2)=O)c(C)nc(=N)[nH]c1C 92034,C1(C(=O)NCCC(CNC(=O)C(C)(C)n2cncn2)OC)CCc2c[nH]nc2C1 92035,C1(CC(=O)NCC(C(=O)OC)OC)CCCN(C(=O)C(OC)OC)CC1 92036,N1(C(C(C2CC2)SC)=O)CCCC(O)(CCNC(=O)CCC2CC2(F)F)C1 92037,N1(C(C2N(CCCC)CCCC2)=O)CCCCC(NC(C2(CC(C)C)CC2)=O)C1 92038,C(=O)(C(CNC(c1c[nH]c(=NC)s1)=O)CC(C)C)NC(CCC)C(C)(C)C 92039,c1(C(C)C)ccc(CC(=O)NCCCNC(=O)C(C)Cc2ccc(Cl)cc2)cc1 92040,C1(NC(C(C)CC(C)(C)C)=O)CN(C(C2CN3CCC2CC3)=O)C2(CCCC2)C1 92041,c1(C(=O)NCC(C)CO)c(Cl)nn(C)c1Cl 92042,c1(CC)cc(C(=O)N(C)CCN2CCN(C(=O)C(O)COC)CC2)ccc1F 92043,C(=O)(C(C)NC(C1CCCC1)=O)N(CCNC(CSCC#C)=O)C 92044,CCC1=NOC(CC(=O)NCCC2CCN(C(C3C(Cl)(Cl)C34CC4)=O)C2)C1 92045,c1(C(C(=O)NC(C)C)N(CCCC)CC2CCC2)ccc(N2CCCC2=O)cc1 92046,c1(C(=O)NC2CN(C(CSCC=C)=O)CC2N=[N+]=[N-])cnc2c(c1)ncn2C 92047,Nc1cccc(C(=O)NC2(CCO)CN(C(c3ccnnc3O)=O)C2)n1 92048,c1(C(N2CC(C)C(C)C2)C(=O)NC(CC)C)c(Cl)nc(Cl)n1C 92049,Cc1ccc(C(CNC(=O)CC(C)(F)F)NC(c2ccn(C3CC3)n2)=O)cc1 92050,C1(CN(CCCNC(c2c(C)onc2)=O)C2CC2)CCC(C)(C)CC1 92051,N1(C(C=Cc2ccc(OC(C)C)cc2)=O)CCN(C(=O)CCCF)CCC1C 92052,C1(CCC(N2C(C)(COC)C=CC2)=O)CCCCN(C(c2cccnc2)=O)C1 92053,C(CCCCC(=O)NC(C1CCOC1)CC)NC(c1n(C=C)ncc1)=O 92054,C1(C(N2CCC(O)(CN(C(CCCC(=C)C)=O)C)C2)=O)Cc2ccc(F)cc2O1 92055,CC(C)C(C(=O)N1CC(CNC(=O)COc2ccc(C(N)=O)cc2)C1)C(C)C 92056,c1(OCCCC(N2CC(C)C(NC(=O)C(C)C(C)(C)O)C2)=O)ccc(F)c(F)c1 92057,N1(C(C(=O)NC2CCCN(c3ncccc3Cl)C2)=O)CCOC2(CCCC2)C1 92058,N1(C(C(C)N(C(COCCC#C)=O)C)=O)CC2(C1)CC(C)(O)C2 92059,n1(CCF)nc(-c2ccoc2)nc1-c1ccc(OCC(F)F)cc1 92060,Cc1ccc2cc(C(=O)NCCCNC(=O)C(F)C3CC3)c(C)nc2c1 92061,N1(C(=O)CSC(F)(F)F)CCN(C(=O)CCC(F)(F)F)C2CCCCC2C1 92062,C#Cc1cccc(C(=O)NCc2cccc(CNC(C3CC=CC3)=O)c2)c1F 92063,C(=O)(CC(C)C(C)C)NC1CN(C(C2(CC)CCCCC2)=O)CC1SC 92064,Cn1cc(C#N)cc1C(=O)NC(CC1CCOCC1)C(=O)NCc1nnc(O)o1 92065,C1(CNC(CCN(C(C)C)C(C2CC3CC(=O)C2O3)=O)=O)CCCC2(CC2)C1 92066,CC(CC(F)(F)F)N(C)C(C1C2CC1N(C(=O)C#CC1CC1)C2)=O 92067,N1(C(CCOC(CC(C)C)C)=O)CCCC1(C)CNC(C1CN(C)C(=O)N1)=O 92068,c1(N2CC(OC)C2)ccc(NC(N2CC(C)(N(C)C)C2)=O)cc1 92069,c1(CC(=O)NC2CC(NC(C(C(C)(C)C)NC(C)=O)=O)C2)c(C)nc(C)nc1O 92070,c1(C(N2CC3CCCCC3C2)=O)ccc2c(-c3ccc(CO)o3)cccc2n1 92071,C1(C(=O)NC(CN(C(=O)C(C)SC(F)(F)F)CC)C)CC2CCC(C1)S2(=O)=O 92072,N1(C(Cc2cn(C)nc2)=O)CCOCC(NCc2cccc(O)c2Cl)C1 92073,C12(NC(C3CCN(C)CC3)=O)CCCN(C(=O)Cc3cc(F)cc(Cl)c3)CC1C2 92074,n1(CC)ncn(NC(=O)C(CCNC(=O)CNC(=O)C(C)CC)C2CCC2)c1=O 92075,c1(-c2nc(C)nn2CC(=O)N(C(C)(C)C)CCN)ccc2ccccc2n1 92076,c1(C(N2CCC(CNC(C3(C=C)CCCCC3)=O)C2)=O)nnn2ccccc12 92077,C(CC(C(=O)O)NC(=O)CCSc1ccccc1)NC(N)=O 92078,C#CC1(F)CN(C(c2ccoc2CNC(C2CC2(C)C(F)F)=O)=O)C1 92079,Cc1c(NC2(C)CCCCCC2)ncnc1N1CCC(C(O)C(N)=O)CC1 92080,CC1C(C)N(C(c2cnc(F)c(F)c2)=O)CCN1C(=O)CCc1cnccn1 92081,N1(C(Cc2cn(NC(c3ccc(Br)cc3)(CC)CC)nn2)CC(=O)OC)CCOC(C#N)C1 92082,C=C(C)C1OCCC1C(=O)NC(C12CCC(CC1)C2)CNC(=O)Cc1cnc(C)s1 92083,N1(C(CCC(C)OC)=O)CCC(C2(NC(c3ccccc3C#N)=O)CCC2)CC1 92084,C(CNC(=O)CC(=O)N(C)CC1(C)CC(C)C1)(CC(=O)Nc1nccs1)OC 92085,c1(C(=O)NC2CCCN(C(C=CC)=O)CC2)cc(S(=O)(=O)NC)cs1 92086,c1(C(=O)NC2C(OC)CN(C(c3c(OC)ccnc3)=O)C2)cc2n(n1)CCO2 92087,C1(C)(C(N(CCCCN(C(C(CC)NC(C)=O)=O)C)C)=O)CCCCC1 92088,C12CCCN(C1)C2=O.C1(C(N(CC(=O)N(CC)CC)CC)=O)CC(C(N)=O)C1 92089,C1(NC(=O)C(F)C2CCOC2)(CNC(C23CCC(C2)C3)=O)CCCC1 92090,C1(CNC(C2CC3(CCOC3)C2)=O)CCC2CN(C(c3ccon3)=O)CC12 92091,C1(C(N2CCCC(N(C(=O)CC3CCCS3(=O)=O)C)C2)=O)CCCCC1(F)F 92092,c1(C(=O)NCC2(CNC(Cc3ccc(C)s3)=O)CCC2)cc2cn[nH]c2cn1 92093,c1(CC)ncnc(N2CC3CC2CN3C(=O)CCc2c(C)c[nH]c2C)c1F 92094,c12ccn3cc(nc3c1)C1(CN(C(CCCCC)=O)C1)COC2=O.N(C)(C)CC 92095,N1(C(c2c(CCC)n(CC)nn2)=O)CCN(C(C2CSC2)=O)C(CC(C)(C)C)C1 92096,Cc1cnc(N(C2CCCNCC2)C(c2ncccc2C)=O)nc1 92097,C1(C(=O)NCCOCCOC)(CC)CCCN1C(=O)C(C)NC=O 92098,N1(C(CC(COC)(C)O)=O)CCN(C(=O)CCOCC2CCCO2)C2CCCC12 92099,c1(CC(=O)NCC2(F)CC(NC(C3CC3F)=O)C2)cc(Cl)ccc1Cl 92100,N1(C(C2(COC)CC2)=O)CCC2(CC2C(N2CC(C#N)(COC)C2)=O)C1 92101,c1(C(=O)NCCCNC(C2(S(N)(=O)=O)CC2)=O)ccc(=O)n(CC2CCCO2)n1 92102,C1(NC(CC2CCC(C)C2)=O)CCCN(C(C2CC3(CSC3)C2)=O)C1C 92103,Nc1nn(CC(N2CCCCC(NC(C3CCCCC3O)=O)C2)=O)cc1[N+](=O)[O-] 92104,C1(C)(CC)CC(C(=O)NCc2cc(C(=O)NC(C)Cc3cnccn3)no2)C1 92105,C(=O)(CC(C)CC(C)(C)C)NC(CC1CC2N(C(CC=CC=C)=O)C(CC2)C1)C 92106,c1(CC(=O)NCC2=CCN(C(COC(C)=O)=O)CC2)c(C)[nH]c2ccnn2c1=O 92107,CN1CCC(CCNC(C2CC(C)(NC(C3CCCCC3)=O)C2)=O)C1 92108,Cc1cc(N)c(F)c(C(N2CCCC(O)(CNC(C3(O)CC3)=O)CC2)=O)c1F 92109,C1(C#N)(C(=O)NCC(CNC(C(C)=C(CC)C)=O)OC)CCCC(=O)C1 92110,C1(NC(c2cc(C)oc2)=O)COC2(CNC(=O)C(C)(C)n3cc(Cl)cn3)CC1C2 92111,c1(C(=O)NCC2(C)CC(NC(C(C3CCCCO3)OC)=O)C2)ccc(Cl)cc1 92112,C(c1ccc(F)c(F)c1)=C(C)C(N1CCC(NC(=O)CCN2CCC2)C(C)C1)=O 92113,C1(NC(C(CC)SC)=O)CCN(C(=O)CCC(C)(C)C#N)CCC1CO 92114,C12(C(=O)NOc3cc(F)c[nH]3)CCN(C(=O)CCc3nccs3)CCC1C2 92115,Cc1cc(=O)n(CCC(N2CC(N(C)C(C3C4COCC34)=O)C(O)C2)=O)cn1 92116,Cc1ccc(C(N2CCN(C(=O)C(C)n3cncn3)CC2C2CCC2)=O)c(N)n1 92117,c1(CC)c(C(=O)N(C)CCOCCCN(C(=O)C(F)CC)C)sc2ccccc12 92118,C(c1csc(Br)c1)=CC(=O)NC1CCCC(NC(=O)CC2CCC2)C1 92119,N1(C(CC2(C)CCCCC2)=O)CC(CO)C2(C1)CN(C(c1ccc(N)cn1)=O)C2 92120,c1(C(=O)NCCN(C(=O)C(C2CCCCCC2)C)CC)cncc(C2CC2)c1 92121,c1(C(=O)NCc2[nH]nc(C(C)(C)O)n2)ncn2c1COc1ccccc1-2 92122,c1(C(=O)O)ccc(CC(=O)OCc2nccn2Cc2ccccc2)cc1Cl 92123,CC1CC(NC(C2(C(F)(F)F)CC(F)(F)C2)=O)CN1C(c1cncc(O)c1)=O 92124,c1(C(CNC(CCSC)=O)N(C(=O)C(C)C2(O)CCC2)C2CC2)ccccc1 92125,C(=O)(C1=CCC(C)(C)CC1)N(CCN(C(c1ccc(OC)cc1Cl)=O)C)C 92126,CC1CCC(C)(C(N2CC(O)(CNC(C3CCCCN3C(C)C)=O)C2)=O)CC1 92127,C1(C(=O)NC2(CNC(CCc3onc(C(C)OC)n3)=O)CCC2)OC2CCC1C2 92128,N1(C(C2(SCC)CC2)=O)CCN(C2CCC(NC(c3cncc(C)c3)=O)C2)CC1 92129,Cc1nc(N(C)C)sc1C(N1CCCC1C1CCCN(C(c2cncs2)=O)C1)=O 92130,N1(C(c2cc(-c3ccc(C)o3)[nH]n2)=O)CCCC1(C)CNC(c1cnccn1)=O 92131,Cc1cc(C(N2CCC(CCC(N3CCN(C(C)(C)C)CC3)=O)C2)=O)n(C)n1 92132,c1(C(N2CC(Cc3cn(CCC(C)=O)nn3)OCC2)=O)cc2sccc2cn1 92133,CC1COCC(CNCC2CCC(C3CC3)O2)O1 92134,c1(C(=O)NCC(CC)NC(c2cnc(OCC)s2)=O)noc(C)c1[N+](=O)[O-] 92135,N1(C(C#CC(C)C)=O)CC(C(=O)NC2CCCN(c3ncccn3)C2)C(C)(C)C1 92136,N1(C(C(C(C)NC(CC(C=C)CCC)=O)C)=O)CC2(CCOC(=O)N2)C1 92137,N#CC1CN(C(c2cnnc(Cl)c2)=O)CCN1C(c1cc(O)cc(O)c1)=O 92138,C1(C2CCCN(C(=O)CCN(C)C)C2)(NC(C2(C(C)(F)F)CC2)=O)CC1 92139,N1(C(c2c(C)nc(C)[nH]2)=O)CC2CCN(C(c3c[nH]cc3C(C)(C)C)=O)CC2C1 92140,c1(CCC(=O)OC(c2ccc(OCCOC)cc2)=O)cncc(OC)c1 92141,CC(C(=O)N1CC(OCC(F)F)C1)C(C)NC(=O)CC1(O)CCCC1 92142,CC1(C)CC(NC(C2(CO)CCCCC2)=O)CN(C(c2ncc(F)cc2N)=O)C1 92143,N1(C(c2n(C)nc(Cl)c2)=O)CCC=C(C(=O)N2CCCC2(C)C2CCC2)C1 92144,c1(C(=O)NCC(C)NC(c2cc3n(n2)CCCC3)=O)cc2nc(Cl)ccc2s1 92145,C12(C(N3CC(NC(c4cc5n(n4)CCO5)=O)C(O)C3)=O)CCC(CO)(CC1)C2 92146,c1(CNC(C2(C3CCCN3C(C3CCCS3)=O)CC2)=O)ccc(O)nn1 92147,C1(CS(=O)(=O)OC)CN(N2CC(O)(CC#N)C2)CC1C(F)F 92148,C1(NC(CCCNC(C=Cc2ncn(C)c2)=O)=O)CC2(CCOC2)C1 92149,N1(CC)CC(C(=O)NC2CN(C(c3ccccc3C(F)(F)F)=O)CC2C)CC1=O 92150,N1(C(c2cc(COC)sc2)=O)CC(CNC(C2CCN(C)C2=O)=O)C(O)C1 92151,N1(C(COCCC(=O)OC)=O)CCc2ccccc2C(NC(=O)C(C)(F)F)C1 92152,c1(C(=O)Nc2cccc(C#N)c2)cnn2c1CN(C(c1n[nH]cc1[N+](=O)[O-])=O)CC2 92153,C=CCC(CC=C)NC(C1CCCC1NC(=O)CN(C)CCC)=O 92154,Cc1nc(C(=O)NCC(C)(O)CNC(=O)CN2CCCCCC2)cc(O)n1 92155,C1(C)(CC(=O)N(CC(C)C)C)CCN(C(=O)COC2CCN(C)CC2)C1 92156,C(=O)(CCc1nccs1)NCCN(C(CNC(C)=O)=O)C 92157,C1(NC(C23CC(C)(OCC2)C3)=O)CN(C(C2CCCS2)=O)CC12CCCC2 92158,C(=O)(C(O)(C(F)(F)F)c1ccccc1)NCC1OCCN(C(CN(C)C)=O)C1 92159,Cn1cc2ccc(NC(C3CC34CCN(C(=O)CCCCCl)CC4)=O)cc2n1 92160,c1(NC(C(C)OC(c2cncc(C(F)(F)F)c2)=O)=O)c[nH]c2ccc(F)cc12 92161,c1(N2CCC(c3ccc(C)s3)CC2)ccc2ncccc2c1[N+](=O)[O-] 92162,CC1CCC(CNS(=O)(=O)c2ccccc2OC(F)(F)F)Cc2ccccc21 92163,c1(C2(C(=O)NCC3(F)CC(NC(=O)Cc4cscn4)C3)CC2)ccc(Cl)nc1 92164,N1(C(CCc2ccc(C)cc2)=O)CC(N(C)C(c2ccnnc2O)=O)C2(CC2)C1 92165,C(=O)(C1=COCCO1)NCC(C(C)C)NC(C(CC=CC)C)=O 92166,C(N=c1ccc(C#N)n[nH]1)C1CCCN(C(c2c(C)ccc(C(N)=O)c2)=O)C1 92167,C1(CNC(C2(CC(C)C)CCCC2)=O)CCCCN1C(c1cncc(N)c1)=O 92168,C1(NC(CSCC=C)=O)CC(C(=O)N(C)CC2CC(F)(F)C2)CC1O 92169,N1(C(CCN(C(C(C)SCCCC)=O)CCCO)=O)CCC(C(=O)NC)CC1 92170,Cc1nc(O)nc(C)c1C(=O)NC1CC(NC(=O)COc2cccc(F)c2F)C1 92171,CCC(CCOC)C(=O)N1CCSCC1CCNC(c1cnccc1C)=O 92172,CC1CC=C(C(=O)NC(C(=O)NC2CC2(C)C(F)F)C(C)(C)O)CC1 92173,C1(NC(C2CN(C)C(=O)N2)=O)C2CC3CN(C(c4ccc(Cl)s4)=O)C1C3C2 92174,C1(N(C(c2c(CC(C)C)onc2)=O)CCO)CCCN(C(c2ccns2)=O)C1 92175,Cc1cccc(C2(NC(N3CCC(CC(C)C)C3)=O)CC2)c1 92176,c1(C(C)=O)ccc(Br)cc1NC(C1CCN(C(c2cc(C)n(C)n2)=O)CC1O)=O 92177,c1(CC(=O)NCCNC(=O)CC2CC(F)C2)cn2c(n1)CCCC2 92178,CC1(C)C2CCC1(C)C2C(N1CCC(O)(CCNC(=O)C(F)=C2CCC2)CC1)=O 92179,CCC(F)(F)C(=O)NCC1(OC)CN(OC)C1.C12CC1(Cl)C(=O)OC2=O 92180,c1(C(=O)NCC2(CNC(C(C(=C)Cl)(C)C)=O)CC23CCC3)nnn2c1CCCC2 92181,c1(C(N2CCC(N(C(CN(c3ccccc3)C)=O)C)C2)=O)cc(O)c(F)cc1N 92182,c1(C(=O)NC23C(CN(C(c4cc(OC)ns4)=O)C2)C3)c(C)cccc1C 92183,C(CC1c2ccccc2CCN1C(c1cc(C)cs1)=O)NC(COCCSC)=O 92184,CN=c1ccc(C(=O)NCCC2CN(C(=O)CN(C)S(N)(=O)=O)C2)c[nH]1 92185,C(C(C)CC(F)(F)F)NC(C(c1ccccc1)NC(c1ccc(C)cc1)=O)=O 92186,C(CCCC(=O)NCC(O)CCNC(=O)CSC1CC1)N(C(C)C)C 92187,N1(C(C(CSC)OC)=O)CCC(C(=O)NCC2CCSC2)=C(F)C1 92188,CCCC(C)(CC)C(=O)NCCN1CCN(C(c2cc(C)n(C3CC3)n2)=O)CC1 92189,N1(C(c2c(COC)cc[nH]2)=O)CC2CN(C(=O)CC(C)(C)OC)CCC12 92190,c1(C(N(C)CC2(NC(C(CCOC)C)=O)CC2)=O)ccc(Cl)c2occc12 92191,C(CO)(C(=O)NCC1CCC(NC(C2CCN2C2CCCC2)=O)C1)N(C)C 92192,C1(CC#C)CCN(C(c2cn(C(C)C)nc2Br)C(=O)NC2COC2)CC1 92193,c1(CCC(=O)NCC2C(C)(C)C2)c(F)cccc1F.C12CC1C(=O)N2 92194,c1(OC)ccc(C)c(NC(C2C=CCN(C(C3(C(C)(C)OC)CC3)=O)C2)=O)c1 92195,c1(C2(C(=O)NCCCCCNC(C(COCCOC)F)=O)CC2)ccnc(Cl)c1 92196,Cc1cccc2c(C(=O)NCC(CC(F)(F)F)NC(C3CC3F)=O)nccc12 92197,c1(CN(C(CC(=O)O)CC2CCCCC2)C2CC2)cc(O)nc(C2CCC2)n1 92198,N1(C(C(C)=CC)=O)CC(C)OC2(CCN(C(=O)CCNS(=O)(=O)CC)C2)C1 92199,C1(C(=O)NCC(CN(C)C(C2(C(F)(F)F)CCC2)=O)O)CC(C)(F)C1 92200,C1(C2CN(C(C)=O)C2)CN(C(C2CC(Cc3ccccc3)=NO2)=O)CCO1 92201,C1(C)(CC)CC(NC(C2(CO)COC2)=O)CN1C(c1cc(OC)cc(Cl)c1)=O 92202,C1(C)(NC(COC2CCN(C(c3c(C)cco3)=O)C2)=O)CC(C)(C)OC1=O 92203,c1(CC)nnc(C)cc1C(N1CCN(C(=O)CCNCCCCOC)CC1C)=O 92204,c1(C(=O)NC(CN(C(c2cnc(S)[nH]2)=O)CC)C)ccc2c(C)cc(O)nc2c1 92205,C(=O)(C(C(C)(C)OC)c1ccccc1)NC(CC)C(F)F 92206,CC(C)CC(O)C(C)C(=O)NCn1ccc(C(=O)NCCC2CC2)c1 92207,CCC(Cc1ccccc1)CC(=O)NC1CN(C(=O)CS(C)(=O)=O)C(C)(C)C1 92208,C1(NC(COCCC)=O)CC(NC(C2CC2[N+](=O)[O-])=O)C(O)C1 92209,C(=O)(C1=CCCOC1)NC(C(CO)NC(c1c(C)sc(Cl)n1)=O)C 92210,c1(OCC(=O)NCC(CNc2cc(SC)ncc2)(C)O)cc(C)cc(C)c1 92211,C(CCCC(C)NC(=O)C(C)Oc1ccccc1)NC(C1(COC)CCCC1)=O 92212,c1(OCC)ccc(C(=O)NC2CCC(N(C(=O)CS(C)(=O)=O)C)CC2)cc1 92213,C(=O)(C1CCc2cccnc21)NCC1(C(C)(C)C)CCN(C(C=COCC)=O)C1 92214,c1(CNC(CC2(C)CCN2C(=O)CC2CCOC2=O)=O)cncc(O)c1 92215,C#CC1(C(=O)NC(c2ccnn2CC)C)CN(C(=O)CC2CC(CC)=NO2)C1 92216,C1(C)(C(N2CC(OC)(CNC(=O)CNC(c3ccncc3)=O)C2)=O)CCCCC1 92217,c1(C(=O)NC(C)CCNC(=O)Cn2nccn2)cn(CC(F)F)cn1 92218,c1(CN(C)CC2C(N3CCN(C)CC3)CCC2)cnc2ccc(Cl)cn12 92219,Cc1csc2ccc(C(=O)NC3CC(CNC(C4CC5CC4C5)=O)C3)cc12 92220,c1(CNC(C2(OCC)CCC2)=O)cc(C(N2CCC(OC)C2)=O)ccn1 92221,C1(N(C(CN2C(C)CC2)=O)C)CCCN(C(c2sccc2C(F)F)=O)CC1 92222,Cn1ccc2cccc(C(=O)NCC3CC(F)CN3Cc3ccccc3Br)c12 92223,C1(CNC(c2cc(F)cc(F)c2Br)=O)CCN(C(c2cn[nH]c2)=O)CC1(F)F 92224,N1(C(C(=C)C)=O)CC(=O)Nc2c(Br)cccc21 92225,N1(C(CC(C=C)CC)=O)CC2CCC1C(CNC(=O)C=Cc1csc(C)n1)C2 92226,CC1(CNC(C2(C#N)CC3CC3C2)=O)CCN(C(=O)COC(F)F)CC1 92227,N1(C(=O)C(c2cccc(I)c2)F)CC=C(c2c[nH]c3ncccc23)CC1 92228,N1(c2ccnc(N3CCCC(C(C)C)CC3)n2)CCc2nncn2CC1 92229,c1(C(=O)NCc2cn(CCCN(C)C(C3CC3(F)F)=O)nn2)cn(C)nc1C(F)F 92230,C1(C)(C(=O)NCC(CNC(C(CC)F)=O)O)CNC(=O)C1 92231,C1(O)(CN(C(=O)C(F)C2CC2)C)CCN(C(C2CN(c3nnnn3C)C2)=O)CC1 92232,Cn1nnc2c1C(C(=O)NCC#CCNC(C1CCOCC1(C)C)=O)CCC2 92233,CC1(C)CCC(n2cc(C3CCOC3)nn2)CN1C(c1ccn2nccc2c1)=O 92234,N1(CC(COCC(c2ccccc2)OC(C)=O)O)CCCC(NC(C)=O)C1 92235,N#Cc1ccc2c(c1)CCCN2C(N1CCC(c2cc(O)nc(=N)[nH]2)C1)=O 92236,c1(OC)cccc(C(=O)NCC(C)N(C(=O)CC2(O)CCCOC2)C)c1OC 92237,N1(C(C(C)NC(=O)C(C)(C)C)=O)CC2CC(C1)CN(C(C1CC1C(N)=O)=O)C2 92238,c1(CC)ncncc1C(N1CCCC1C(C)(C)NC(=O)C(C)Cn1ccnc1)=O 92239,c1(C(=O)NCCN(C(=O)CCCCC(N)=O)C(C)C)ccc2[nH]cc(C#N)c2c1 92240,c1(COC)cnc(OC)c(C(=O)NC2CC(OCC(C)C)C2(C)C)c1 92241,CC1(C(=O)NCCc2ccsc2)CCCN(C(c2c[nH]c(=N)o2)=O)C1 92242,N1(C(C(N2CC(C)C2)C)=O)CCN(C(c2ccncn2)=O)CC1c1nccn1C 92243,Cc1cc(CN2CCN(c3ccc(C4CC4)c(C)n3)CC2)ccc1F 92244,C1(C(N2CC(CC=C)(NC(c3c[nH]nc3SC)=O)C2)=O)CCOC1C=C 92245,N1(C(C2CCCO2)=O)CC2(C(=O)NC(CO)C(F)(F)F)CC1CO2 92246,C1(CC=C)(NC(=O)CN(C)CCO)CCCN(C(C2CC2F)=O)C1 92247,C(=O)(C(O)CCCc1ccccc1)N1CC(C)C(NC(=O)CC(C)(C)C)C1 92248,C(=O)(CCCS(C)(=O)=O)NCC1(CNC(C(C)Cc2cnco2)=O)CC12CCC2 92249,C=CC(C)(C)CC(=O)NCCOC1CN(C(C2CCC(C)S2)=O)C1 92250,C(C)(C)(CC(F)C(=O)N(C)CC1COC(=O)N1)NC(c1c(C)c[nH]n1)=O 92251,C(=O)(C(C)(C)C(C)O)N(CC=CC(N1CCC(C)(NC(C)=O)C1)=O)C 92252,C(N=c1nnc(C)c(C)[nH]1)C1(C)CCN(C(c2ccc(N(C(C)=O)CC)o2)=O)C1 92253,c1(OC)cc(F)c(Cl)cc1C(=O)NC1CN(C(C2CC(F)(F)C2)=O)CCC1O 92254,c1(C(=O)NC(CC=CC)C(=O)Nc2cncnc2OC)c[nH]c(=N)c(C)c1 92255,N1(c2cc(N3CCC(NC(n4ccnc4)=O)C3)ncn2)CCCOC(C(F)F)C1 92256,CC(C)C(C(=O)NC1CC(C)(C)C12CC2)C(C)NC(=O)CCCn1ccnc1 92257,C1(C(=O)Nc2cn(CC=C)nc2)CC(C)CN(C(=O)CCn2cnnc2)C1 92258,N(C(=NCc1nc(C2CC2)n[nH]1)NC1CCCC(CF)C1)Cc1sccc1 92259,c1(-c2c(C(=O)NCC3C(NC(c4cc(C)no4)=O)CC3)c[nH]c2)ccccc1Cl 92260,c1(C(=O)NCC(C)=CC(=O)NC(CN(C)C)C(C)(C)C)cc(C#N)ccc1N 92261,C1(NC(C2C(OC)CN(C(CCC#CC)=O)C2)=O)CC2(CCCC2)C1 92262,c1(OCC(=O)NC(CN(C(c2c(C(C)C)nco2)=O)C)C)ccccc1C#N 92263,Cc1cccc(N2CCN(C(c3ocnc3C)C(=O)NCC3CCOC3)CC2)c1 92264,C1(C(N2CC3C(CC(=O)NCc4nc(C)c(C)s4)C3C2)=O)CC2(CCC2)CO1 92265,C1(CNC(c2scc(C(N)=O)c2)=O)C(O)C(O)CN1C(C1CCCCC(=O)N1)=O 92266,C(C(O)C(C)(C)C)NC(C(C)NC(Cc1c(C)ocn1)=O)=O 92267,N1(C(c2c3c([nH]n2)C(C)CC3)=O)CCOC2(C1)CN(Cc1ccc(O)cc1F)C2 92268,C=C(C)CCN(CC(C)NC(=O)NCC)C 92269,CC1CC(NC(c2ccsc2)=O)CN1C(=O)CC12COCC(C1)C2 92270,Fc1cc(Cl)cc(Br)c1OCCN1CCC(Oc2ncc3cn[nH]c3n2)CC1 92271,C1(CC(N2CC(NC(c3coc(C4CCC4)n3)=O)C(O)C2)=O)CC2(CCC2)CO1 92272,c1(CC)cc(C(=O)NCC(O)CCNC(C2CCSC2)=O)cc(C)c1 92273,C(=O)(CC1=CCCCC1)NC1C(C)(CN(C(CC2(OCC)CCC2)=O)C)CCC1 92274,C1(OC)CC2(CCCN(c3cc(N4CCN(C(=O)C5CC5)CC4)ncn3)C2)C1 92275,C#Cc1cc(C(=O)NCC2(C)CCCN2C(=O)CCC2CC2(C)C)ccc1Cl 92276,C1(CCCNC(C(C2CC(C)(C)C2)OC)=O)CCCCN1C(=O)C=CCO 92277,C12(C(N3CCC(N(C)C(c4nn(C)nc4C(F)(F)F)=O)C3)=O)CNCC1COC2 92278,c1(NC2CCC3CN(C(c4c(C(C)C)ccs4)=O)CC32)ccc([N+](=O)[O-])cc1F 92279,c1(C(N2C(CN(C)C(C3CCCC3(F)F)=O)CCC2)=O)c[nH]ccc1=N 92280,N1(C(C=CC(C)(C)C)=O)CCc2c(CNC(=O)CC34CCCC3C4)cccc2C1 92281,C(=O)(C(CN(C)C)CC)NCc1c(C(=O)NC(C(=O)OCC)C)[nH]cc1 92282,C(=O)(C(C)S(C)(=O)=O)NCc1c(C(N(C(c2nccs2)C)C)=O)n[nH]c1 92283,N1(C(C2(OC)CC2)=O)CCCC2(CC(NC(=O)C=C3CCC(C)CC3)CO2)C1 92284,C1(C2CC2)(CNC(C2(OC)CCC2)=O)CCN(C(c2c(Br)nnn2C)=O)C1 92285,Cc1nc(C(N2CC(F)CC2CNC(C2C(C(F)F)C2(C)C)=O)=O)cn1C 92286,CC(C)CC(F)C(=O)NCCC1CCCCN1C(c1ccnn1C(C)C)=O 92287,c1(CNC(=O)COCCNC(C2CCCS2)=O)ccncn1 92288,N1(C(CC(C)c2ccccc2)=O)CC(O)CC1C(=O)Nc1nc(C(F)(F)F)cs1 92289,C#CC1(O)CN(C(=O)CSCCNC(C2(CF)CC2)=O)C1 92290,CC#CCCC(=O)N1CC(OCC)C(NC(=O)CCCN(C)C(C)C)C1 92291,C1(O)(CN(C(=O)CCC2CCC(=O)N2)C)CN(C(=O)CCc2cnoc2)C1 92292,c1(SCC)ccc(C(=O)NC(C)(C)CCCNC(=O)Cn2cc(C#N)cn2)cn1 92293,C1(CC(=O)NCC(C)(CO)NC(C(C)=C2CCC2)=O)COC(C)(C)C1 92294,C=C1CCN(C(c2cc(Cl)n(C)n2)=O)C(C(=O)NCCOCCN=[N+]=[N-])C1 92295,C1(NC(C(COC)(F)F)=O)COC2(CNC(=O)C(c3cccs3)SC)CC1C2 92296,C#CCC(CC(F)F)C(=O)N1CCCC1CCC(=O)Nc1ccc(C)cc1CO 92297,CCC(CC)CC(F)C(=O)N1CCC2(CC1)CC2C(=O)Nc1cccc(O)c1F 92298,N1(C(c2ccc(CC)cn2)=O)CC2(C)CC1(C(N1CC3CCC3(CO)C1)=O)C2 92299,c1(C(=O)NCC(C)NC(CC2CC(OC)C2)=O)ccc(N2CCCC(O)C2)cc1 92300,C(C1=CCN(Cc2cc(Cl)ccc2Br)CC1)NC(c1cccc(F)c1C1CC1)=O 92301,C1(C(N(CCNC(C2(OC)CCCC2)=O)C(C)C)=O)C2CCN(CC2)S1(=O)=O 92302,N1(C(C(C)OCC=C)=O)CC(C(N2CCCC(C(C)(C)O)C2)=O)C(C)(C)C1 92303,N1(C(C2(OCC)CCC2)=O)CC2(CC(C(=O)NCCn3ccnc3C)CO2)C1 92304,C=CCCCCCCC(=O)N1CCN(C)C(CNC(=O)CC2CC(OC)C2)C1 92305,c1(OCC)c(NC(C2CC2(C)C(F)F)=O)cc(F)cc1Br 92306,C1(S(C)(=O)=O)(C(=O)NC(C)CC(C)NC(c2ccncc2F)=O)CCC1 92307,c1(C(=O)NCC(CNC(C2(c3ncco3)CC2)=O)OC)cc(F)c(F)cc1F 92308,C(=O)(CC(C)C(=O)NC1(C)CN(C(=O)CCn2cc(Cl)cn2)C1)OC 92309,Cc1nc(C2CC2)[nH]c1C(=O)NCC1(CCNC(C2(C)CCCC2C)=O)CC1 92310,N1(C(C2CC=C(C)CC2)=O)CCCC2CN(C(=O)CC3CC=CCC3)CC12 92311,N1(C(C(=O)N(C)C)=O)CCN(C(c2cccc3c2NCC3)=O)C2CCCCC12 92312,Cc1ccc(CC(N2CC(CNC(=O)CNS(N)(=O)=O)C(O)C2)=O)c(F)c1 92313,CCC(CCC(=O)N1CC(n2cccn2)C1)NC(=O)CC(C)C1CC1 92314,CC1CCN(C(=O)C(=O)NCC(F)F)C1CNC(c1c(Br)ncn1C)=O 92315,C(=O)(C(C)S(=O)(=O)C(C)C)NC(CC(C)C)CNC(=O)CCc1cnn[nH]1 92316,N1(C(C(C)=CC)=O)CC(CNC(=O)CC(CC)CCC)OC2(CCC2)C1 92317,c1(N(C)Cc2ccccc2[N+](=O)[O-])ccc(S(=O)(=O)NCC2CCCCS2)cn1 92318,C(CCCC(=O)NCCCCCO)N(C(C1C(C(C)C)OCC1)=O)C 92319,C1(CC(=O)N(C2CCN(C(=O)COCCF)CC2)C)COC(C)(C)CO1 92320,N1(C(C=CC(=O)N(C)C)=O)CCOC2c3ccccc3OCC12 92321,C1(NC(C=C(C)C(F)F)=O)CCCN(C(C2CCC2(F)F)=O)CC1 92322,O1NC(=O)C(F)C2(O)CN(C(=O)C1(C)C)C2.c1(OC)ccc(=N)[nH]n1 92323,CC1CN(C(C2CCCN2c2cnccn2)=O)CCN1C(=O)C=CBr 92324,C1(NC(CCn2c(C)cc(C)n2)=O)CN(C(C2CCC2C)=O)C2(CCC2)C1 92325,C1(CC(=O)N(C)CC2N(C(C3CC(OCC)C3)=O)CCOC2)COCC(C)(C)O1 92326,N1(C(COCCCC)=O)CCN(C(C2(C)CCC(OC)C2)=O)CC12CCC2 92327,C1(C)(N(C(c2cncc(-c3c(C)nccc3)n2)=O)C)CCS(=O)(=O)C1 92328,C1(CNC(C(C)CC2CCC2)=O)CCCN(C(c2c(C(F)(F)F)cnn2C)=O)C1 92329,C1(CNC(C2C(C=C)C2)=O)COCCN1C(=O)CC1CCSCC1 92330,c1(C(N2CC(C)N(C(=O)Cc3c(Cl)cnn3C)CC2)=O)cnn2c1N(C)CC2 92331,O=C(C=Cc1ccccc1F)NNc1ccc(Cl)cc1F 92332,C1(NC(C=CC=CC)=O)CC2COCC(C1)C2NC(=O)CC1CCS(=O)(=O)C1 92333,C1(C(N2CCN(CCNC(=O)CC3=CCCC3)CC2)=O)CC2CCCCN2C1 92334,c1(C(=O)N(C2CC(C(=O)NOC3CCCCC3)C2)CCO)c[nH]c2cccnc12 92335,Cc1nc(C(=O)N(C)C)ncc1NC(=O)C=Cc1ccsc1C(F)(F)F 92336,C1(CC)CCN(C(c2cc(OC)n[nH]2)=O)C1CNC(=O)C(CCSC)OC 92337,C1(CNC(C(c2cccc(O)c2)C)=O)CCN(C(=O)C=CC2CCCC2)CC1 92338,CCC(C)(CC)CN=c1[nH]c2c(c(=NCC(=O)NC3CC3)[nH]1)CCCCC2 92339,c1(C(=O)NC(CN(C(c2cc(CN(C)C)c[nH]2)=O)CC)C)c(Cl)cnn1C 92340,c1(CCC(=O)NCC(F)CNC(C2(C(F)F)CC2)=O)ccc(F)c(Br)c1 92341,c1(C(C)C(=O)NC(C2(O)CN(C(c3ncccc3Cl)=O)C2)C)c(F)cccc1F 92342,C(=O)(C(CCF)N(C(=O)C(CCC)NC(N)=O)C)NC(C=C)C 92343,c1(C(=O)OC)coc(C=CC(=O)NCC(C2CC2)NC(=O)Cc2ccon2)c1 92344,N1(C(CC=C)=O)CCN(C(c2csc(N(c3ccccc3)C)n2)=O)CC(C)(C)C1 92345,c1(C(=O)NC2(C)CC(NC(C3(C)CCCS3)=O)C2)ccc2nc(C3CC3)[nH]c2c1 92346,C1(C(=O)NCC(=O)N(C(c2ccncc2)C)CC)CCC(OC)CC1 92347,Cc1ncnc(C(=O)NC2CCCC2C(=O)NCC2(F)CCOC2)c1C 92348,c1(OC)n[nH]c(C(=O)NC2(CNC(=O)CC3(O)CCCOC3)CCCC2)c1Cl 92349,N1(CCN=C(NCC(CC)CO)NC2CCC2)CCc2ccccc21 92350,C1(CNC(C(C=C)O)=O)CC(F)CN1C(C1CCC(C)O1)=O 92351,C(=O)(CC1=CCN(C(c2c(F)cccc2F)=O)CC1)Nc1ccc(C)nc1C 92352,c1(C(N2CC=CC(NC(C3(CC=C)CCOCC3)=O)C2)=O)onc2ccccc12 92353,c1(C(C)N(C(=O)C(C)(C2CC2)N(C(=O)CN(C)C)C)C)ccccn1 92354,N1(C(CCOC)=O)CC(Cn2cc(C(O)C(C)(C)C)nn2)C(C(F)(F)F)C1 92355,C(=O)(CCCCC(C)CC)NC(CCCC)CNC(c1ncoc1C(F)(F)F)=O 92356,C1(NC(CCCSC)=O)CCC2CN(C(c3ncoc3C(C)(C)C)=O)CC2C1 92357,C(CC(F)CN=[N+]=[N-])NC(c1cc(CNC(C(C)NC(CC)=O)=O)ncc1)=O 92358,Cc1nn(CC(N2CCCC(N(C(=O)CO)Cc3ccccn3)C2)=O)c(C)c1C 92359,C1(C(N(C(CC)C2CC2)C)=O)COCCC1NC(c1cc(C)sn1)=O 92360,c1(N(C)Cc2cnn(CC)c2C)ncnc(NC2CC3CCCC3C2)c1C 92361,c1(CC(=O)N(C2CCN(C(C3CCCS3(=O)=O)=O)C2)CC)c[nH]c2ccccc12 92362,Cc1ccc(Cl)c(N)c1C(=O)NCCC(O)CNC(C12CCN(CC1)C2)=O 92363,CCCC(CCCNC(=O)CSCCC(C)C)NC(c1coc(CC)n1)=O 92364,c1(OC)ccc(C(N2CC(CNC(=O)CC3CCOCC3)CC2(C)C)=O)c(F)c1 92365,CCC(O)CC(=O)NCCC1(CNC(=O)CCc2nc(-c3ccco3)no2)CC1 92366,CC1(C)CC(NC(C2(C)CCCC2(F)F)=O)CCN(C(c2cc(N)ccn2)=O)C1 92367,C1(CNC(=O)CC2CNC(=O)C2)CCN(C(C2CC2[N+](=O)[O-])=O)CC1 92368,c1(NCCCN(C)C(C23CC4CC(C(=O)N2)C3C4)=O)ncnc2c1nnn2C 92369,Cc1c[nH]c(C(=O)NCC2(CCNC(c3ccoc3C3CC3)=O)CC2)cc1=O 92370,C(CCC(C)C)(C(=O)NCCOCCN(C)C)NC(C(CC)n1cncn1)=O 92371,c1(CC)cccc(NC(c2sccc2CNC(c2n[nH]cc2C)=O)=O)c1C 92372,C1(C(N(CC(=O)N(C)C)CCC)=O)CCCN(C(=O)C2=C(Cl)CC2)C1 92373,c1(C(=O)NCC2CC(NC(C(c3n(C)ncc3)O)=O)C2)ccc2c(c1)COC2 92374,c1(C(=O)NC(C2(C(=O)NC3CCCC3(F)F)CC2)C)ccc([N+](=O)[O-])o1 92375,C=CC1CN(C(c2cccc[n+]2[O-])=O)CC1NC(c1ccc(C(C)C)c(F)c1)=O 92376,c1(C(=O)NC(C(C)NC(Cc2ccc(OC)cc2)=O)C(C)C)c(F)cccc1F 92377,C1(CCC(=O)NC)CCCN1C(=O)N(C)CCO 92378,c1(C(N2CCN(C3(S(C)(=O)=O)CC3)CC2)C)ccc(Cl)cc1 92379,CCC(CC(=O)N1CCC1CNC(C1(OC)CC1)=O)c1ccccc1 92380,C1(O)(COC)CCN(S(=O)(=O)CC2CCCCO2)C1 92381,c1(NC2C(NC(c3cnn(-c4ccccc4)c3)=O)CCC2)cccc(Br)c1I 92382,c1(C(=O)NCC(C)(O)CNC(C2CC2(Cl)Cl)=O)cn2ccccc2n1 92383,c1(NC(C)CN(C(C(C(C)C)SC)=O)C)c(F)cccc1[N+](=O)[O-] 92384,c1(C(=O)NCC(C2CCCCC2)NC(C(C)OCCOC)=O)ncc(Cl)cc1Cl 92385,c1(OC)ccc(Cl)c(F)c1C(=O)NCC(C(C)C)NC(=O)CSc1ccncc1 92386,c1(OC)ccnc(NCC(=O)NCC(C)CNC(C2(C)CCCC2C)=O)n1 92387,C1(C(F)F)(OC)CCCN(C(c2nc(Br)nn2C)C(=O)NC(C)(C)C)C1 92388,N1(C(C(C(C)C)C)=O)CCn2ncc(CNC(C3C4CCOCC34)=O)c2C1 92389,Cc1c(C(=O)NCCC(C)CCNC(=O)C(C)C2(O)CCC2)cccc1Cl 92390,C1(NC(c2c(C)nsc2)=O)C(C)CN(C(=O)C(C)(C)COCC(F)F)CC1C 92391,c1(C(=O)NC(CN(C(CCC(CCCC)C)=O)C)C)cc(F)c2nc(C)cn2c1 92392,CCCCC(O)C(=O)NCC1(C)CCN(C(c2cccnc2OC)=O)C1 92393,c1(CCC)ccc(F)cc1C.C1C(CC(C)C)S1 92394,C(CO)(CC(C)(C)C)NC(C1C(CNC(Cc2nc(C)[nH]n2)=O)C1(C)C)=O 92395,C1(C(=O)NCC2(C=C)CCC2)C2CCCC2CN1C(C1CCC2(CCC2)C1)=O 92396,C(C(CNC(C1CCS(=O)(=O)C1)=O)S(C)(=O)=O)NC(C1(CC#C)CC1)=O 92397,c1(C(N(C2CCN(C(C(C)NS(C)(=O)=O)=O)C2)C)=O)cc(Cl)c(Cl)[nH]c1=N 92398,C=C=CCC(=O)N1CCC(C(C)(C)NC(c2cc(C(C)CC)no2)=O)C1 92399,C(C(CC(=O)N1CCC(CO)(NC(=O)C2=CCOC2)C1)C(F)(F)F)N(C)C 92400,N1(C(c2coc3c2COC3)=O)CCN(C(=O)C(F)(F)C(F)(F)F)CC2(CC2)C1 92401,CC(C)CCC(=O)C(=O)N1CC(C2CC2C(N2CCC(CCCO)C2)=O)C1 92402,C1(O)(CNC(c2cn(CCNC(CCC=C(C)C)=O)nn2)=O)CCC(C)C1 92403,C#CCC(C)C(=O)N1CCN(CCCNC(c2cc(CN(C)C)on2)=O)CC1 92404,c1(OCCCC(=O)NC(CNC(C(C)OCOC)=O)(C)CO)ccccc1Cl 92405,CC(CC(=O)N1CCC(O)(CNC(=O)CC2CN(C)C2)C1)C(F)(F)F 92406,c1(SC)cc(C(N2C(CNC(=O)CCC3CCCCO3)CC3CC23)=O)ccc1F 92407,C(C1CCCO1)=CC(=O)NCC1CCCC1NC(=O)CC(O)c1ccccc1 92408,C(=O)(CCCN=[N+]=[N-])NCCCCC(C)NC(C1(CCOC)CC1)=O 92409,CCC(C(=O)NCCCCC1(NC(=O)Cc2csc(Cl)n2)CC1)C(F)(F)F 92410,CC(C)(C#N)CCCC(=O)NCC1C(CNC(c2c(F)cccc2F)=O)C1(F)F 92411,C1(NC(c2csc(C(F)F)c2)=O)CC2CN(C(c3ccccc3)=O)CC12 92412,C12(C(=O)NC(C)(C)C)CC1CCCN2C(=O)O.N12CCC(C1)N(C)C(=O)C2.CN 92413,c1(C(=O)OC)cc(CN2CC(NC(c3scc(C)c3C)=O)C2)cc([N+](=O)[O-])c1 92414,C1(CCNC(C=CCC)=O)C(C)CCCN1C(c1cc(OC)ncn1)=O 92415,Cc1cc(C(N2CCC2C(=O)NCC2CCOC2)=O)oc1C 92416,N1(C(C2CC(C)N2C(C2CC3CCC(C2)O3)=O)=O)CCc2ccccc21 92417,N1(C(COC2C(CC)CCCC2)=O)CCC2(CCCN2C(C2CC3(CC3)C2)=O)C1 92418,c1(C(N2CCC(C(CO)NC(c3c(C)onc3)=O)CC2)=O)ccc2nonc2c1 92419,C1(NC(C2(COC)CCC2)=O)CN(C(=O)COc2cccc(F)c2)CC2(CC2)C1 92420,C1(C(=O)OC)CCS(=O)(=O)C12CN(C(=O)C(=O)NC1CCN(CC(F)F)CC1)C2 92421,c1(C(N2CCCC(N3CCCC3=O)C2)C(=O)NCC(C)C)cnn(C(C)C)c1I 92422,C1(C(=O)NC(c2ccc(C)nc2)C)CCN(C(c2ccccc2F)=O)C(C)(C)C1 92423,C(=O)(C1=CCc2ccccc21)NC(C)CC(C)NC(c1cnc(Cl)n1C)=O 92424,C(c1c(F)cccc1F)=CC(=O)NC(CC)CNC(c1ccc(C(N)=O)[nH]1)=O 92425,C1(NC(CCC(N)=O)=O)CCC2CCN(C(=O)C(C3CC(F)(F)C3)O)C1C2 92426,N1(C(C(CC(C)C)=O)=O)CCC2CN(C(C3(C4CC4)CCC3)=O)CC2CC1 92427,n1(CC)cnc2c(NC(c3nc[nH]n3)C)[nH]c(=NCc3nncs3)nc12 92428,N1(C(C(c2ccccc2)OC)=O)CCCOC(CNC(C2(SC)CC2)=O)C1 92429,c1(C(N2C(C)CC(CNC(CCSC)=O)C2)=O)cc2n(n1)CCCNC2=O 92430,n1(CCCC=C)cc(C(=O)NCC(C)CNC(=O)COCc2nc[nH]n2)nn1 92431,N1(C(C2C(C)(C)CO2)=O)C2CCC1CN(C(C1CC3C=CC1C3)=O)C2 92432,C1(N(C(C(CCC)CC)=O)C)CC2CCC(C1)N2C(=O)C(F)(F)C(O)CC 92433,c1(N(CCC)CCNC(C2(C#N)CCC2)=O)cc(N2CCNC2=O)c(F)cc1F 92434,c1(C(=O)NC2C(OC)CN(C(c3cccnn3)=O)C2)ccc(F)c(CO)c1 92435,C1(O)(C(=O)NCCCC2(NC(Cc3ccn(CC)n3)=O)CC2)CCC(C)(C)CC1 92436,Cc1ncc(CCNC(=O)CCN(C(=O)C=CC2CCOC2)C(C)C)[nH]1 92437,N1(C(C(CC)(F)F)=O)CC2CCN(C(=O)CCC3CC3(Cl)Cl)CCC2C1 92438,c1(C(C(N2C(C)(CNC(COC(CC)C)=O)CCC2)=O)=O)ccc(Cl)cc1O 92439,c1(C(=O)NCCC(C)Nc2cccc(F)c2[N+](=O)[O-])coc2c1C(O)CCC2 92440,c1(OC)cc(F)ccc1C(=O)NC1CCN(C(=O)Cc2cc(C)nn2C)C12CC2 92441,CC1CN(C(=O)Cc2cc(O)nc(O)n2)CCN1C(c1coc(Cl)c1)=O 92442,c1(CNC(c2n(C)nc(C(=O)OCC)c2NC)=O)cnc2ccc(Br)cn12 92443,c1(C(=O)NCC2CN(C(CC3(C=C)CC3)=O)CC2O)nc2n(c1Cl)CCCC2 92444,c1(C(=O)NCC2(NC(c3ccsc3)=O)CC2)cccnc1-n1ccnc1 92445,N1(C(C(C)=CC)=O)CCCC2(C1)C(NC(c1cc(F)n[nH]1)=O)CCN2C 92446,c1(C(=O)NCC(CC)(C)NC(c2csc(COC)c2)=O)nc(O)sc1C 92447,N1(C(C2C(C)CCC2)=O)C2CCC1CN(C(=O)C=Cc1ccncc1)C2 92448,c1(C(N2CCN(C(C3CC34CCC4)=O)CC2CCO)=O)ccc([N+](=O)[O-])c(Cl)c1 92449,C1(C(=O)NC(CC)(C)C(F)(F)F)CCN(C(=O)CN(C)C2CC2)C12CCC2 92450,C1(C(=O)NC2C(CNC(CNS(NC)(=O)=O)=O)CCC2)COC(C)(C)CO1 92451,Cc1cccn2c(CC(=O)NC(C)C(=O)NC(c3ccccc3)C(=O)O)cnc12 92452,c1(NC)cc(Cl)ccc1C(N1CCC(CO)C(NC(C2(C)CCCCO2)=O)C1)=O 92453,CCCCCC(C)NC(=O)C(c1cnn(C)c1)NC(c1ccc(F)s1)=O 92454,C1(C(=O)NCC2(OCC)CC2)CSC(CCC(C)C)C(=O)N1 92455,CCC(=O)CCC(=O)N1CCCN(CCNC(=O)Cn2cccn2)CC1 92456,N1(CCN(C)C)CCN(C(c2ccc3c(c2)CC3)C(=O)NCCC2CC2)CC1=O 92457,c1(C(=O)NCCC2CC(C(=O)NCC3(C)CCCO3)C2)cnn2c1OCC2 92458,C1(CC(=O)NC2CCN2C(=O)COCCOc2ccccc2)CCCCC1(F)F 92459,Cc1cc(C(=O)NCC2CC2NC(=O)Cn2ccc(C3CC3)n2)ccn1 92460,c1(C(=O)NCC2N(C(c3c(C)nns3)=O)CC=C2)cnc2nc(O)ccc2c1 92461,N1(C(CC2CCC(C)C2)=O)CC23CCCC2(C1)CN(C(c1coc(CO)c1)=O)C3 92462,c1(C(C(N2C(C(=O)OCc3ccccc3)CSC2)=O)O)cc(F)c(F)cc1F 92463,C1(C(=O)NCc2ccn(C(C)C)n2)CCCC(NC(c2c[nH][nH]c2=N)=O)C1 92464,c1(CCNC(C(C2(C)CC2)NC(C(C)=CCC)=O)=O)ccn(C)n1 92465,CN1CCN(C(=O)C(F)(F)c2cnccn2)CC1CNC(C1(C)CC=CCO1)=O 92466,c1(CNC(C(=O)NCc2ccc(SC)cc2)=O)ccc2c(c1)CCO2 92467,Cc1cc(C(=O)NCCC2CC(NC(=O)Cc3ccsn3)C2)n2nc(C)cc2n1 92468,N1(C(CC2CC(=O)C2)=O)CC(NC(=O)C=CC(F)(F)F)C2CC12 92469,CC1(C#CC(=O)NC2CN(C(=O)C3=CCCCC3)CC23CC3)CC1 92470,Cc1onc(CC(=O)NC2CCC(CNC(C3CCCC(O)C3)=O)CC2)c1C#N 92471,CN1CCC(CNC(C2CC(NC(c3ccncc3)=O)CCO2)=O)CC1 92472,N1(C(CC2CCCN(C)C2)=O)CCC2(CCC2CNC(=O)CCC2CC2)CC1 92473,C1(NC(Cn2c(C)ncc2)=O)CN(C(C2(Cl)CC2(C)C)=O)CC(C)(C)C1 92474,C(F)(F)(C(=O)NNC(=O)COC(C#N)C1CC1)c1cccc(C)n1 92475,N1(C(c2cc(C(F)(F)F)cc(Br)c2)C(=O)NC(C)C)CCCC2CC(C)CCC12 92476,N1(C(C(C)(C)C2CC2)=O)CC2(C=C(C(=O)NOCCCCN3CCCC3)CO2)C1 92477,C1(NC(c2cccc(C)c2Cl)=O)CN(C(c2cc(O)cc(Br)c2)=O)CCC1(F)F 92478,c1(C(=O)NCC(CCNC(c2cc(C(F)F)nn2C)=O)OC)cc(C)nc(N)c1 92479,C1(CNC(c2ccc(Cn3cc(CC4CCCC4)nn3)o2)=O)CCCOCC1 92480,C1(CNC(C2(C)CCN(C)C2)=O)CC2(CC(NC(=O)CC3CC4(CCC4)C3)C2)C1 92481,C1(SC)CN(C(=O)CSc2nncs2)CC1NC(C1CC(C)C1)=O 92482,C1(NC(C=Cc2ncc(C)[nH]2)=O)CN(C(=O)C(C2CC2)C2CC2)CC1C1CC1 92483,N1(C(C23CN(C(CCC)=O)C(C2)CO3)=O)C2CCC1CC(C(C)C)C2 92484,c1(N(C(CCNC(C2(OC)CCS(=O)(=O)C2)=O)C)C)ccc([N+](=O)[O-])cc1Cl 92485,N=c1nc2c(c[nH]1)CC(C(=O)NCCCCNC(=O)CC13CCCC1C3)CC2 92486,C1(CC(=O)NCC(C2CC2)NC(c2cncc(C=C)c2)=O)CCC2(CCC2)CO1 92487,C1(C(N(CC(CNC(CCC#C)=O)O)C)=O)CC(c2cn(C)nc2C)=NO1 92488,C12CCCCN(C1)C(=O)C1CCCN1C(=O)C(=O)N2C.C1(N(C)C)(CC)CC1 92489,CC1(C)NC(=O)N(CC(=O)NC2CC(NC(=O)C(CO)NC(N)=O)C2)C1=O 92490,C1(C(N(CC(=O)Nc2nnc(-c3ccccc3)s2)C)=O)CCCN2CCCC12 92491,c1(C(N(C)CC2CN(C(C34CC(F)(C3)C4)=O)C2)=O)cc2n(n1)CCNS2(=O)=O 92492,c1(C(N2CCC(C)(NC(C(CC(C)C)NC(N)=O)=O)C2)=O)cnn2c1NCCC2 92493,C1(NC(Cc2c(C)con2)=O)CCCCN(C(=O)C(F)C(C)(F)F)C1 92494,c1(C(=O)OCC)cnn(C)c1S(=O)(=O)NCC1OC(=O)CC1(C)C 92495,Cn1ncc([N+](=O)[O-])c1C(N1CC2CC(C1)C2O)=O 92496,N#Cc1c(NC(C2CCN2CC(=O)NCc2ccc(Br)o2)=O)cccc1Br 92497,C1(OC)CCC2CN(C(=O)CC=CCNC(C3(CO)CCC3)=O)CC12 92498,C#CC1(C(=O)NC(c2ccc(O)nc2)C)CCN(C(C2C=C(C)CS2)=O)C1 92499,C1(CC)C(C(=O)NC(c2ncc(F)cn2)C)CCCN1C(C1CCC1COC)=O 92500,C(C(C)(C)C(=O)NCc1ccc(C(N2CC(OCC(C)C)C2)=O)nc1)SC 92501,Cc1cc(F)cnc1C(=O)NC(CC1CC1)C(=O)NCC1CC2(CCC2O)C1 92502,N1(C(C=C(C)C)=O)CCC(N(C(c2cnco2)=O)CC2CC2)C1 92503,C1(OC)CN(C(=O)COC2(C)CCCC2)CC1CNC(C1CCCN1N=O)=O 92504,C(N=c1cc(C)nc(C)[nH]1)C1CN(C(c2cc(C)ncc2)=O)C(C)C1 92505,C1(C(N2CC(CC)(NC(=O)Cc3cccnc3O)C2)=O)CCC2CC1C2(C)C 92506,C(CC1CCc2ccccc21)NC(N1CCCC1Cc1cc(F)ccc1Cl)=O 92507,C1(NC(C2N(C(CCC)=O)CCCC2)=O)CCN(C(=O)CCCC(F)F)C1(C)C 92508,c1(C(N(CCCNC(=O)CC(C)(C)F)C(C)C)=O)cc(Cl)cc(F)c1N 92509,C1(CC)CC(C)CN(C(C2CCC(CNC(=O)CCCC3CC3C)CC2)=O)C1 92510,C=C=CC(C)C(=O)NC1CCN(CCNC(=O)C(C)CC=C)CC1 92511,c1(C(=O)NCc2cn(CCOC(C)=O)nn2)ccc(-n2cc(Br)cn2)cc1 92512,C=CCC(CC)C(=O)N1CC(NC(=O)CCSCC(C)C)CC1(C)C 92513,c1(C(=O)NCC(C)NC(C2CC2(F)F)=O)ccc2c(c1)B(O)OC2 92514,c1(C(=O)NCC(CC(C)C)NC(c2ccn(C)c2)=O)cc2ccc(Cl)c(F)c2[nH]1 92515,N1(C(C(C2CCCO2)OC)=O)CC2(CCN(C(c3cc(N)c(F)cc3C)=O)C2)C1 92516,N1(C(CCc2ccn(C)c2)=O)CCN(C(=O)CNS(=O)(=O)N(C)C)C(CCO)C1 92517,c1(-c2nc(SCC(C(C)C)N(C)C)n(CCOC(C)C)n2)nccn2nccc12 92518,C(=O)(CC1OCCc2ccccc21)N1CCC(C)(NC(=O)CC2(O)CCC2)CC1 92519,C(=O)(C(COC(C)=O)C(F)(F)F)NC1C2(NC(C(CCCC)C)=O)CCC(C1)C2 92520,Cn1ncc(C(=O)NC2CCN(C(=O)CC3CC(C)(C)C3)C2)c1-n1cccc1 92521,N1(C(CC2(NC(C3C4CCCCC34)=O)CC2)=O)CCC2(CCO2)C1 92522,c1(CC)ccc([N+](=O)[O-])cc1C(=O)NC1CCN(C(C2CSCC(=O)N2)=O)CC1 92523,CC(CC(=O)NC1(C)CCN(C(c2ncccc2O)=O)C1)C(F)(F)C(F)(F)F 92524,N1(C(C2CN(CC)C(=O)C2)=O)CC2(CCN(C(c3ccc(Cl)o3)=O)CC2)C1 92525,N1(Cc2ccc(C#C)s2)CC2(CN(C(=O)Nc3ccccc3F)CCO2)C1 92526,c1(OCC(=O)NC2C(NC(c3c(Br)ccc(C)c3)=O)C2)ccc([N+](=O)[O-])cc1 92527,c1(C(N2C(C)C(C)N(C(c3cncnc3)=O)CC2)=O)ccc(S(=O)(=O)CF)cc1 92528,CC1C2CC(C2OC(C2CN3CCN2CC3)=O)N1Cc1ccccc1 92529,C1(CN(C(c2c(C)cns2)=O)C)CN(C(=O)CCc2cccc(O)n2)CCO1 92530,c1(OCC)cc(F)c(C(=O)NCCC2CN(C(=O)C=CC3CCOC3)C2)c(F)c1 92531,c1(CNC(C(=O)N(C(C)CNC(=O)CCN(C)CCO)C)=O)ccc(F)cc1 92532,N1(C(c2nc(OC)nc(O)c2)=O)CCOC2(C1)CN(C(=O)C(F)n1ccnc1)C2 92533,C(=O)(C1CNCc2ccc(Cl)cc21)N1CCC2(CC(CC(=O)O)OC2)C1 92534,C(=O)(CC(C)(O)C(F)(F)F)N1CCN(C(CSCC#C)=O)CC1CO 92535,N1(c2snc(C)n2)CC2(COC(CNC(C3CC4(CCCC4)C3)=O)C2)C1 92536,C1(NC(c2ccccc2)CC)CCN(C(C2CC23CCC3)=O)CC1C 92537,C1(c2ccccc2)(CNC(COC(C)=O)=O)CCN(C(=O)CC2(C)CC2F)CC1 92538,c1(CCC)cc(C(N2CC(N(C(=O)CSc3nccn3C)C)C2)=O)n(C)n1 92539,c1(CNC(CN(C2CC(C#N)C2)C(C=C(C)C(F)F)=O)=O)csnc1C 92540,c1(NC(C2C(NC(CCCn3c(C)ncc3)=O)CCC2)=O)cc(Cl)ncc1Br 92541,N1(C(CCC=C(C)C)=O)CCC2CN(C(C3CC34CCCC4)=O)CCC12 92542,C#Cc1cn(C)nc1C(=O)NC1CCCCC1CC(=O)NCC(F)(F)CO 92543,c1(CNC(C2N(C(C3CC(OCC)C3)=O)CCC2)=O)ccc(O)c(C)c1 92544,c1(C(C)NC(=O)NC2CC(C)(COC)C2)cccc(SC)c1 92545,C1(C(=O)NC2C(C)(C)CN(C(=O)Cc3ccsc3)C2)CCc2nccn2CC1 92546,C#Cc1ccc(C(=O)NCCC(C)NC(C2CC(C#N)C2)=O)c(F)c1 92547,C(c1cnc(O)nc1O)=CC(N1CC(NC(C2CC23CC(O)C3)=O)C2(C1)CC2)=O 92548,N1(C(C2(CC)CC2)=O)CCN(C(c2ccc(C3CC3)c(F)c2)=O)CC12CCC2 92549,CCC(C)C(O)C(=O)N1CC(CN(C)C(c2ccnc(C)c2)=O)C1 92550,CC1(CC(=O)NCC2CN(C(=O)Cn3nccn3)C3CC23)CCOCC1 92551,c1(CC)cccc(CNCC2(F)CC(COC)C2)c1OC(C)(C)C.O 92552,c1(OC)cc(C)ccc1NC(C1CC1(c1ccccc1)F)=O 92553,NC1CCN(C(c2csc(-c3ccc(Br)s3)n2)=O)C(C(F)(F)F)C1 92554,N1(C(C2CCN(CC)CC2)=O)CCN(C(C2CCSCC2)=O)C(CC#N)C1 92555,N1(C(C(C(C)C)SCC)=O)CCOC2(CCN(C(=O)CCCc3cncs3)C2)C1 92556,C(C(F)(F)CCNC(C1CCN(S(C)(=O)=O)C1)=O)n1cc(CN(C)CC)nn1 92557,C1(NC(c2nc(C)n(C)n2)=O)CC2CC(NC(=O)C3=CCOCC3)CC2C1 92558,Cc1cn(-c2cccnc2)[nH]c1=NC(=O)NC1CCN(CC(F)F)C1 92559,C1CCN(C(c2csc(C)n2)C)C1.C1(C)(C(=O)NN2CCCC2)CCCS1 92560,CC1Oc2c(C(=O)NC(CNC(=O)C(C)(F)F)C3CC3)cccc2NC1=O 92561,O=CN1CCOCC1C(N1CC2CC2(CNC(C2CC(C3CC3)=NO2)=O)C1)=O 92562,N1(C(C(C2CCS(=O)(=O)CC2)(C)C)=O)CCN(C(=O)C2=CCCOC2)CC(O)C1 92563,C1(C(N2CCC(N(C(=O)C=CSC)CCC)C2)=O)CCc2nc(C)ncc2C1 92564,c1(OC)ccc(N(C(c2ccc(OC)cn2)C(=O)NC2CC2)CC(F)F)cc1 92565,Cc1cc(CNC(=O)NC(Cc2cccc(Br)c2)C(=O)O)ncn1 92566,C(C(C)(C)CN=c1[nH]c(=N)[nH]c(=NC(C)c2nc(Cl)ccc2Cl)[nH]1)OC 92567,c1(C(=O)NC(C2CCN(C(C3(OC)CCCOC3)=O)CC2)C)cnc(Cl)cc1N 92568,c1(C(=O)OC)cc(S(=O)(=O)N(C(c2ccccc2)CF)C)ccc1F 92569,C1(NC(Cc2c(C)occ2)=O)CCOCC1NC(C1(CCO)CC1)=O 92570,C=C(C)C(C)(O)C(=O)NNC(=S)Nc1ccc2ccccc2c1 92571,Cc1ncnc(C(=O)NC(C)CC(C)NC(=O)CCC(=O)c2ccc(Cl)s2)c1C 92572,c1(C(C(N2CC(C)OC(C)C2)=O)(C)C)ccc(Cl)cc1[N+](=O)[O-] 92573,C(=O)(C(CC(C)C)N(C1CC1)CC1CC1)OC.c1(C2C(=O)N2)ccccc1Br 92574,CC1CN(C(=O)C(C)(CO)NC(c2ccc(C(N)=O)o2)=O)Cc2nncn21 92575,N1(C(C(C(C)C)N2CCCC2=O)=O)CC2CCCN(C(c3cc(O)no3)=O)C2C1 92576,N1(C(C(CC2CC2)OC)=O)CCC(O)(CCNC(C2CC(F)C2)=O)CC1 92577,c1(C(=O)NCC(=CC(=O)NC(C(CCC)C)CO)C)ccc2cc[nH]c2n1 92578,c1(NC(CC2(C)CN(Cc3c(OC)c(F)ccc3)C2)=O)nccc2[nH]ccc12 92579,c1(C(N2CC(NC(C3CCCC(F)(F)C3)=O)C(F)CC2)=O)ccc2c(c1)COC2 92580,Cc1cccc(C(=O)C(=O)Nc2cccc(CNC(=O)CC(C)C)c2)c1 92581,c1(C2CO2)cn(C(C)(C)C(C)C)nn1.C(COC)(OC)OCCN(C)CCOC 92582,CP(C)(=O)c1ccc(C(=O)NCC23CCCC(CN2C(=O)COC2CC2)C3)nc1 92583,N1(C(=O)CCCC(F)F)CCC2(CCN(C(=O)C3=CCCC3)C2)C1 92584,N1(C(c2ncnc(C)c2C)=O)CCCC2(CCN(C(=O)COCC(F)(F)F)C2)C1 92585,c1(C(N2CCC(C(C)(C)NC(C(F)OC)=O)C2)=O)cccc2ccc(O)nc12 92586,C1(CS(C)(=O)=O)CCCN1C1CN(C(c2nnc(Br)s2)=O)C1 92587,C1(C(=O)NC(C(=O)NCC(=O)OCC#C)CCSC)CC(=O)C12CCC2 92588,c1(CC(=O)NCC(c2ccccc2)NC(c2cc(C)sc2)=O)c(C)noc1Cl 92589,Nc1ncnc2c1ncn2CC(=O)Nc1cccc2c1ncn2CC(F)(F)F 92590,c1(CCC)nc(C)c(C(=O)NCCC2CC(NC(=O)C=CC3CCCC3)C2)o1 92591,c1(CC(=O)NC(C)CCCNC(C2(C)CC2C)=O)ccccc1Br 92592,c1(C(=O)NC2C(C(=O)NCCn3ncc(C)c3)COC2)cncc(F)c1 92593,C(=O)(C(C)C(C)NC(=O)CCN(CCCO)C(=O)Cc1cnns1)OC 92594,CC(C(=O)N(C(C)CCNC(c1ccc(C2CCOC2)cc1)=O)C)C(C)(F)F 92595,C1(C(=O)NCC)CCCN1C(c1ccc(CNC(=O)CCCNC(N)=O)s1)=O 92596,C1(C)(CNC(C2C(C(=O)OC)C2)=O)CCCN1C(=O)COC1CCCCC1C 92597,n1(CC)ccc(C(=O)NCC2CCN(C(=O)CC3(CO)CCCCC3)C2)c1C 92598,C1(C(=O)NCC2C(NC(CCN(C)CC)=O)CCCC2)CCC2CCCCN12 92599,C#CCCCCC(=O)N1CCN(C(=O)CC(C)c2ccccc2)CC1CCO 92600,C(CC(CC)C(=O)NC(C1CC=CCC1)C(=O)NC1CCCC(CO)C1)=CC 92601,S(=O)(=O)(c1c[nH]c(C(N2CC(CCNC(=O)C(O)C(C)(C)C)(OC)C2)=O)c1)NC 92602,N1(C(C(CC)(C)F)=O)CC(NC(c2ccc(CO)nc2)=O)C(N=[N+]=[N-])C1 92603,C1(C(=O)NC2CC(NC(c3ccccc3CO)=O)CC2O)(OC)CCC(C)(C)C1 92604,Cc1cc(C(=O)NCc2ccc(C(=O)NCC3CCCCC3(C)C)s2)nc(C)c1 92605,N1(C(c2c(OC)csc2)=O)CCCC(CC(=O)N(C2CCCCC2O)C)C1 92606,C(=O)(C1=CC2(CCN(C(c3ccc(C(C)C)o3)=O)C2)C1)NCc1ccc(SC)o1 92607,c1(C(=O)NC2(CCF)CCN(C(C)=O)C2)cnc2[nH]c(C(F)(F)F)nc2c1 92608,c1(NC(C2N(Cc3cccc(C#N)c3)CCSC2)=O)ccc(Br)cc1[N+](=O)[O-] 92609,c1(C(=O)NC2CCC(CNC(COCCCC)=O)C2)cc(OC)cc[n+]1[O-] 92610,C1(NC(CN(c2ccccc2)C(C)=O)=O)COCC1C(=O)NC(c1ccsc1)C 92611,C1(NC(c2c(C)snc2)=O)CCCC(C(=O)NCC(O)CNC(N)=O)CC1 92612,c1(CC)nn(C)c(OC)c1C(c1nnnn1C1CCC1)NCC(C)CCO 92613,N1(C(C2N(C(C3(CC)CC(C)(C)C3)=O)CCCC2)=O)CC(C2CCCCC2)C1 92614,c1(C(N2CCC(N(C(c3cnc(O)n3C)=O)CC)C2)=O)cccc2nccnc12 92615,c1(OC)ncccc1C(=O)Nc1cccc(CNC(=O)Cc2c[nH]nc2O)c1 92616,N1(C(C(CC)=CCCC)=O)CC(NC(C2(COC)CCCC2)=O)C(COC)C1 92617,N1(C(CS(CC)=O)=O)C2CCC1C(CNC(c1c[nH]cc(Cl)c1=O)=O)C2 92618,N1(C(CC)=O)CCC(NC(CN(C(C2CC2CC(C)(C)C)=O)CCO)CC)C1 92619,N1(C(CCCCCC)=O)CC2CCCC2(NC(c2nnccc2C)=O)C1 92620,CCC(C)C(=O)N1CCC(NC(c2occc2COC)=O)C1 92621,c1(CC)ccc2[nH]c(C(N3CCN(C(=O)C(F)=C(C)C)CC34CC4)=O)c(C)c2c1 92622,C=CCCN=C(NCC(C)C(F)(F)F)NCc1ccc(C2CC2)cc1 92623,C1(C(N(C)CC2CCCN2C(=O)C2=CCCO2)=O)CC2CCC(C1)N2C 92624,CCC(C)(C(=O)N1CCC(F)(C(=O)NC(C)C(C)(C)C#N)C1)OC 92625,c1(CN2CCN(C(CC(CC)C)=O)C3C2C3)cc(C#N)ccc1Cl 92626,C1(C(=O)NC(C)C(C)(C)NC(c2cncc(Cl)c2)=O)OCCOC12CCC2 92627,Cc1ncc(C(F)(F)F)cc1C(=O)NCC1CCC1NC(c1ccon1)=O 92628,CCC(CC(=O)NC1CCC(NC(c2conc2C2(C)COC2)=O)CC1)OC 92629,c1(C(=O)NCC(CC=C)NC(=O)C2=CCOCC2)cnc2c(Br)cccn12 92630,N1(C(c2cn(CCCC)nc2C)=O)CCOCC(NC(C2(F)C3CCCC23)=O)C1 92631,C(=O)(CCCC(=O)N(CCCOCCNC(=O)C(O)Cn1cncn1)C)N(C)C 92632,c1(C(c2nnnn2C)NCc2c(C(=O)OC)cc(Br)o2)cc(F)cc2c1OCC2 92633,N1(CC(=O)NCC2CCC(NC(C=C(C)Cl)=O)CC2)CCCCC(O)C1=O 92634,N1(C(C=NOC)=O)CC(NC(c2cnc(C)c(C(F)(F)F)c2)=O)CC(O)C1 92635,C1(CC(=O)NCCN(C(C)C)C(C23CC4CC2C3C4)=O)CCCN(C)C1 92636,CCC(C)(C)CCC1CC1C.C1CO1.C1CNC(=O)O1.C1CNC(=O)N1 92637,C1(CC)C(C(=O)NCc2nc[nH]n2)CCCN1C(C1CC2(CC2)CO1)=O 92638,n1(CC(=O)N(C)CC2N(C(C(C)N(C)C)=O)CCC2)ccc2ccccc12 92639,Cn1cnc2c1CCC(C(=O)NC1CC(NC(=O)Cc3ccc(O)c(F)c3)C1)C2 92640,C12(C(N(CC(C)CNC(=O)C(N3CCN(C)CC3)C)C)=O)CC(C)(C1)OC2C 92641,C1(C(=O)NCCCNC(=O)OC)C2CCC(C2)N1C(C1CC2CC2C1)=O 92642,C1(C(N2CC(O)(CN(C(C3C(C(=O)OC)C3)=O)C)C2)=O)C(C)(C)C1(C)C 92643,N1(C(C(=O)NCC2N(S(C)(=O)=O)CCC2)=O)CC2CCC1C1CNCC21 92644,C1(NC(C(CC2CC2)NC(CC2OCC(C)(C)C2)=O)=O)CCCN2CCCC12 92645,Cc1ccccc1C(C)CC(=O)N1CC(O)(C(C)NC(c2nncn2C)=O)C1 92646,Cc1cccc2c1CCOC2C(=O)Nc1ccc(F)c(C#N)c1Cl 92647,CC1CC(CNC(=O)CCC2CC2C)CN(C(=O)C=Cc2ncc[nH]2)C1 92648,CC(CF)CC(=O)N1CCC(C(C)CNC(c2ccn(C3CCC3)n2)=O)CC1 92649,c1(N(C)C)nccc(C#N)n1.C12CCCN(C1=O)C2=O 92650,c1(OC)cc(NC(C2CC2NC(c2cccc(O)c2O)=O)=O)ccc1C 92651,CC(CCCCN=c1c(C#N)c[nH]c2cc(F)cc(F)c12)NC(=O)C1=CCCO1 92652,Cc1cc(F)ccc1C(N1CCOC(CNC(=O)C=CCOCC(F)(F)F)C1)=O 92653,C1(C(=O)NCc2c(C(=O)NCCC3CCN(C)C3)scc2)CCC(=O)NC1 92654,Cc1c(C=CC(=O)NCCCCC(C)NC(C23CCC(CC2)CO3)=O)cnn1C 92655,C(C(C)(CC(C)C)NC(C1CCOCC1(C)C)=O)NC(c1cccc(C)n1)=O 92656,N1(C(CCSC)=O)CC2CCCC(CNC(=O)CN3CCn4nccc43)C2C1 92657,C(C)(C)(CC(=O)N1C(C(=O)NCC2CCC2(F)F)CCC1C(C)C)OC 92658,S(=O)(=O)(c1c[nH]ccc1=NCCC1CC1C)N(CCCCOC)C 92659,N1(C(C2C(C)CC=CC2)=O)CCN(C(=O)CCn2ccccc2=O)CC1CCO 92660,n1(CC)ccc(=NC(=O)C2(C(C)C)CCN(C(c3ncc[nH]3)=O)C2)[nH]1 92661,N1(C(C(C(C)OC)NC(c2cc(=O)n(C)cn2)=O)=O)Cc2n[nH]cc2C1CO 92662,c1(C(=O)NC(CC)CN(C(=O)C(O)C2CC2)C)[nH]c(O)nc1C 92663,Cc1nc2sccn2c1C(=O)NCC(O)CNC(C1C2CCC1CC2)=O 92664,C12(NC(C3CC(OC)C3)=O)CC(CNC(C3(C)CCCC3)=O)(C1)OC2C 92665,C(=O)(CC(C)C(F)(F)F)N1CCCC(CC=C)(NC(=O)CCC=CC)C1 92666,N1(C(CC2OCCN(C(C(C3CCOCC3)C)=O)C2)=O)CCC2(CCCO2)C1 92667,C1(C(N2CCC(C)(CNC(=O)C3=NNC(=O)C3)C2)=O)CCc2nccn2C1 92668,S(=O)(=O)(c1ccc(Br)cn1)N1CC2CCN(C(C(=O)c3ccco3)=O)C2C1 92669,Cc1c(C(N2CCC(C)(NC(=O)CN3CC4CC4C3)C2)=O)cnn1CC(F)(F)F 92670,C1(CC(=O)NC(CCOC)CNC(=O)C(C)(C)C)CCCCCCC1 92671,C1(C(N2CC(C)C(CNC(=O)C(C)S(N)(=O)=O)CC2)=O)CN(C)CCN(C)C1 92672,c1(OCC)cccc(C=CC(=O)NC(c2ccccc2)CNC(=O)C=NOC)c1 92673,C(=O)(CCS(C)=O)NCC1(C(C)NC(c2nc(C(=O)OC)oc2)=O)CC1 92674,N1(C(CCS(C)(=O)=O)=O)CCC2(C1)CN(C(C1CS(=O)(=O)CC(=O)N1)=O)CCO2 92675,N1(C(c2ccc(C)nc2C)=O)CC2CCCC2C1C(=O)NCCCC(F)F 92676,C1(NC(C(N2CCCCC2=O)C)=O)CC12CCN(C(=O)CSc1cccs1)CC2 92677,C(=O)(C(C)(O)C(C)(C)C)NC(C)CNC(=O)Cc1ccc(CO)cc1 92678,N1(C(c2[nH]c(=NC)sc2)=O)CCCOC(CNC(=O)Cc2ccc(Cl)nc2)C1 92679,CCC(CCOC)C(=O)NC1CC(CO)N(C(c2ccc(CC(C)C)cc2)=O)C1 92680,N1(C(CN(CCOC)C)=O)CC2(CCCC2)C1C(=O)NC1(C2CCCCC2)CC1 92681,CC(CC(=O)NC1CC2CSCC2C1)C(C)(C)NC(=O)C=CC(=O)N(C)C 92682,C1(NC(c2cc(C)sn2)=O)CC(NC(c2ccsc2C)=O)C12CCC2 92683,CC1(C)CN(C(C2CCOC2C2CC2)=O)CCC1NC(C1(CCN(C)C)CC1)=O 92684,C1(NC(C2CN(C(c3cccs3)=O)CCO2)=O)CC2CC(O)C1C2 92685,Cc1cc(C)c(C(N2CCC(CCNC(C3CC34CC4(F)F)=O)CC2)=O)cc1C 92686,C1(C(=O)NC2C(SC)CCC2)CCC(O)CN1C(=O)Cc1nonc1C 92687,C1(CNC(CN(CC(C)C)C(C2CC2(C)C(F)F)=O)=O)CNC(=O)CO1 92688,CC1CCCC=C1C(=O)N(C(CC(F)F)C(=O)N1CCC(C(F)F)CC1)C 92689,N1(C(c2ccc(C)o2)=O)CC2COCC(C1)C2NC(C1CCC2(CC1)CC2)=O 92690,N1(Cc2c(C)c[nH]c2)CC2(CN(C(c3cnn[nH]3)=O)C2)C1 92691,C12(C(=O)NC(CC#C)CO)CC1CCN2C(c1nccs1)=O 92692,C(=O)(CCC(CC)CCCC)NCC1C2(CCN(C(C=CC)=O)CC2)C1 92693,C1(C)(C(=O)NCC2C(CCC)C2)CCN(C(=O)COC2CC2)C1 92694,c1(C(N(c2ncc(C(=O)OC)s2)CC)=O)c(C)cc(C)cc1C 92695,C(c1ccccc1F)=CCC(=O)NC(C1N(C(C(CCOC)C)=O)CCC1)C 92696,CN1CCC(CC(=O)NC2(C)CCN(C(C3CCOC3)=O)C2)C1=O 92697,N1(CCOC)CC(C(N2CCC(NC(=O)CCSCC(C)C)C2)=O)CCC1=O 92698,CC1OCCOC1C(=O)NC1C=CC(C(=O)NCCc2ccsc2)C1 92699,C1(CC(=O)NCCC(CNC(=O)CCOc2ccccc2)O)CCCC(=O)N1 92700,C1(CCCC)CCN(C(C2(C)CCN2C(=O)OC(C)(C)C)=O)CC1 92701,c1(C(=O)NCC(CNC(c2c(CC)sc(=N)[nH]2)=O)(C)O)cnc2ncnn2c1C 92702,C1(CC(=O)OCC)CN(C(C)C(N2CCC(N3CCCCC3)CC2)=O)CCO1 92703,N1(CCCCC)CCCC(c2nc(-c3ccc(OC)nc3)nn2C(C)C(C)C)C1 92704,CC(C)(C#N)CCC(=O)NC1CCN(C(c2cc(Br)c(F)cc2F)=O)C1 92705,C1(O)(CC(=O)NCC2CCC2)CCN(C(c2cc(F)cc(F)c2)=O)CC1 92706,N1(C(CC(=O)OCC)=O)CCCN(C(=O)CNC(=O)CC2CCCC2)C(CO)C1 92707,c1(C(=O)NCC(C(C)C)NC(C=CC=CC)=O)cc2c([nH]1)CCC(C)C2 92708,C1(CC(=O)N(CC(=O)OCC2CCCSC2)CC)CCCCN1C(C)=O 92709,Cc1ccc([N+](=O)[O-])cc1NC(=O)NCC(c1ccc(Cl)cc1)O 92710,N1(C(c2ncn(C)c2)=O)CCC(C2(NC(c3cccc(C(C)(C)C)n3)=O)CC2)C1 92711,C1(C)(CC)C=C(C(=O)NC2(C(=O)NCC(C)(CO)OC)CC2)C1 92712,CC1(C(N2CCN(CCNC(C3CC(CF)C3)=O)CC2)=O)COC(=O)N1 92713,C(c1ccc(C)cc1C)=CC(=O)NC1CN(C(C2=CC(C)(CC)C2)=O)CC1F 92714,C1(C(=O)NCC(CC)NC(=O)C=CCN2CCCC2)(CC)CC1(F)F 92715,CCCCCS(=O)(=O)NC(c1cncc(-c2nn[nH]n2)c1)=O 92716,Cc1cc(N)c(F)c(C(=O)NC(CNC(=O)Cc2ccc(Cl)cc2F)CO)c1F 92717,Cc1cc(C(=O)NCCC(C)NC(C2COCCN2CC2CCC2)=O)ncc1F 92718,C1(C(=O)NCCC2N(C(C34OCC(C)(C3)C4)=O)CCC2)CCC(=O)NC1 92719,c1(C(N2CCC(O)(CC(=O)NCC3(O)CC(C)(C)C3)C2)=O)ccc(F)c(F)c1 92720,C(=O)(C#CC1CCCCC1)N1CC2N(C(c3nccc(C)c3)=O)C(CC2)C1 92721,C1(NC(C2(C(=O)NC)CCC2)=O)CCC(NC(=O)CC2CC(F)C2)C1 92722,N1(C(COCCC)=O)CCC(O)(C(C)NC(c2cnc(N(C)C)c(Cl)c2)=O)CC1 92723,c1(CC(=O)OC(C2CCOCC2)C(=O)OC)ccc(OC)nc1C 92724,c1(C(N2C(C)C(NC(c3ccnc(O)c3)=O)CCC2)=O)ccc2ncccc2n1 92725,Nc1ccc2ccccc2c1-c1ccccc1Cl 92726,c1(OC)cc(C)ccc1NC(=O)C(=O)NC1(CO)CC(C)C1 92727,c1(C(N2CCC(F)(CNC(C3(O)CCOC3)=O)CC2)=O)n[nH]c2c1CCCCC2 92728,N1(C(COCCNC(=O)CN2CCOC2=O)=O)CCN(C2CC2)C(=O)C1 92729,CC1CN(C(=O)CSc2nnc(S)s2)CC(C)C1NC(c1cccc(=O)o1)=O 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92835,c12ccc(cc1)NS(=O)(=O)C2.O(NC(=O)COC)CC 92836,C1(C(=O)NCCC(=O)NCC2(NC(CCOCCN(C)C)=O)CC2)CCCOC1 92837,Cc1ncncc1C(=O)N1C(N)CCC1.C1(C(=O)NC)CN(CCC2CCC(C)CC2)CC1O 92838,C(=O)(C(C)(C)C(=O)NC(C(=O)Nc1c(CC)cccc1CC)C(C)C)OCC 92839,C1(CN(C(C(c2ccccc2)OC)=O)C)CCN(C(c2nc(Cl)sc2C)=O)CC1 92840,c1(C(N2C(CNC(C(CCCC)O)=O)CC(F)(F)C2)=O)cc2c(=O)[nH]ccn2c1 92841,N1(C(c2n(CC)ncc2)=O)CCN(C(=O)C(c2cccc(Cl)c2)SC)CC12CC2 92842,C1(C(N(C(C)CNC(=O)CSC(F)F)C)=O)CC12CC(O)C2 92843,c1(NC)scnc1C(N1CCC(C(C)C(=O)NCC(CSC)OC(C)=O)C1)=O 92844,CC(C(=O)NC1CC(C(F)F)(NC(C2COC(=O)N2C)=O)C1)C(F)F 92845,N1(C(CC(C)(C)c2cn(-c3ccc(C)c(F)c3)nn2)=O)CCC(S(=O)(=O)C(C)C)C1 92846,c1(OC)ccc(C(N2CCC3C(NC(=O)C(N)=O)C23)=O)cc1OCCCl 92847,N1(C(C(CC)O)=O)C2CCC1CC(NC(c1cccc(N)c1C)=O)C2 92848,N1(Cc2cn(CCNC(C(C3CC3)OC)=O)nn2)CCCC(N(C)C)C1 92849,c1(C(N2CC(NC(c3cc(CC)on3)=O)C2)=O)c(Cl)cc(C)cc1Cl 92850,N1(Cc2nc(CCOC)on2)CCC2(NC(=O)CC3CCCC(=O)N3)CCCC12 92851,CN=c1nc(NC2CCCn3nc(C)nc32)[nH]c(=NCC(C)c2ccsc2)[nH]1 92852,c1(OC)ccc(Br)c(C(=O)NCC2CCN(C(C3CNC(=O)C3)=O)CC2)c1 92853,c1(N(C(C#C)C)C)nnc(C2CCCCO2)n1CCOCC1CCCO1 92854,C1(NC(C2(COC)CC2(F)F)=O)CCCCC1NC(=O)C(CCO)N(C)C 92855,N1(C(C(C)OCC=C)=O)CC=CC(C(=O)NCC2CCOC2(C)C)C1 92856,CCC(C)C(C(=O)N1CC=CC1(C)C(=O)NCCc1cn[nH]c1)N(C)C 92857,C(=O)(CCCCCCn1cc(-c2csc3nccn23)nn1)NCCC1(C)CCO1 92858,c1(C(=O)NCCN(C(=O)Cc2csc(Cl)c2)CC)ccc(-c2cc[nH]n2)s1 92859,N1(C(=O)CCOc2cc(F)ccc2F)CCC2(CCN(c3cnc(F)cn3)C2)C1 92860,Cc1cccc(C(=O)NCC(C2CCCC2)NC(c2cnn[nH]2)=O)c1C 92861,Cc1sc(Cl)nc1C(N1CC(CC(C)NC(=O)C(C)Cn2cccn2)C1)=O 92862,N1(C(c2cncc(C)n2)=O)CCC2CCC12CNC(c1sccc1OC(F)F)=O 92863,C1(NC(CC(CC)C)=O)COC2(CCN(C(C3CC4CCC3O4)=O)CC2)C1 92864,C1(C)(NC(C(C2CCOCC2)C)=O)CCN(CCOc2cccnc2)C1 92865,c1(C(=O)NC2(CNC(c3csc(Cl)n3)=O)CCOC2)cccc(F)c1O 92866,C1(C(=O)NCC2CCN(C(c3cnc(O)s3)=O)C2)(CF)CC(F)(F)C1 92867,C=CCCCC(C(=O)NOCCCCF)NC(=O)CC1CC=CCC1 92868,C(=O)(C(C)(C)C(C)C)NCC(C)(C)NC(CC(=O)NCC(=O)NC(COC)C)=O 92869,CC1(C)C(C(c2nnnn2C2CCCC2)NCCn2ccnn2)C1(C)C 92870,CCN=C(NCC(c1ccc(Br)cc1)F)NCC1(C2CC2)CCCO1 92871,c1(C(=O)NCCC(C)(C)NC(=O)OC(C)(C)C)ccc(C(F)(F)F)cc1C#N 92872,C1(C2CC2)(C(N2C(CC(N)=O)CCC2)=O)CN(C(c2ncn3c2CCC3)=O)C1 92873,c1(C(N2CC(C(N)=O)(CNC(C3(F)C(C)OCC3)=O)C2)=O)scc2c1CCCC2 92874,O=S(=O)(c1c[nH]ccc1=NC1CCN(c2ccc(Cl)cc2)CC1)NCCCO 92875,C1(CNC(=O)Cc2sccc2F)COCCN(C(=O)CCCc2cccnc2)C1 92876,C1(NC(c2ccn(C)c2)=O)CCCC2CN(C(c3cc(F)n(C)n3)=O)CC12 92877,c1(CC)c(C(N2CCOCC2CNC(C2(C)CC=CCC2)=O)=O)cnn1CC 92878,C12(NC(C3C(CNC(Cc4cc(C)no4)=O)CCC3)=O)CCCN(CC1)C2 92879,c1(N2CCN(C(C)=O)CC2)nc2c(F)cc(F)cc2c(=NC(C)c2nc[nH]n2)[nH]1 92880,C(CNC(C1CC2CC2C1)=O)(CC(F)(F)F)NC(CSc1n[nH]c(=N)s1)=O 92881,N1(Cc2cccc(OC)c2C)CC2CN(C(c3ccc(N(C)C)nc3)=O)CC2C1 92882,C12(C(=O)NCC3(CNC(=O)C=Cc4cncs4)CCCC3)OCCCC1C2(F)F 92883,C1(NC(c2n(C)c(Cl)cn2)=O)CCN(C(c2c(F)cccc2Cl)=O)CC12CCC2 92884,c1(NC(=O)NC)ccc(F)c(C(=O)OC)c1.c12cc(nc(SC)n1)S2 92885,N1(C(=O)Cc2ccccc2)CCCC(c2cn(Cc3ccccn3)nn2)C1 92886,C(c1ccccn1)=CC(=O)NCCC(=C)CNC(=O)CC(C)c1ccncc1 92887,C12(C(=O)NCC(CNC(c3c(CC)n(C)nc3)=O)(C)O)CCC(C1)S(=O)(=O)CC2 92888,c1(NC2CCN(C(C3CCCC(C)C3)=O)C(C)C2)ncnc2c1ncn2C1CC1 92889,N1(C(C(=O)NCCOC)=O)C2CCC1CC(NC(C1CC(=O)N(C3CC3)C1)=O)C2 92890,Cc1[nH]nc(C(N2CCCC(NC(c3ccnc(C(N)=O)c3)=O)C2)=O)c1Cl 92891,c1(C(N2CCCC(NC(C3(CC=C)CC3)=O)C2)=O)c[nH]c2cc(Br)ccc12 92892,CC1=CCSC1C(=O)N(C1CCN(C(c2cnc(Cl)[nH]2)=O)C1)C 92893,CCC1=NOC(C(N2CCC(C(C)(C)C(=O)NCCCc3nccs3)C2)=O)C1 92894,c1(COCC)nc(C(=O)NC(C)CC2CN(C(c3cc(Cl)cs3)=O)C2)cs1 92895,N1(C(C)=O)CC2CCC2(CCN(C(=O)COC2CCCC2)C2CC2)C1 92896,O=C(C1=CS(=O)CCC1)NCCCN1CCN(C(=O)C(F)=CCCF)CC1 92897,N1(C(C(C2CC2)OC)=O)CCN(C(c2cc(C)nc(C)c2)=O)C(C2CC2)C1 92898,C(=O)(CC(C)CNC(=O)C(C)(C)CC1CC1)NC(c1ncc(C)o1)C 92899,N1(C(=O)NC2CC2c2ccc3c(c2)CCC3)C2CCC1CC(C(=O)NC1CC1)C2 92900,C1(C)(NC(C(N2CCC(C)C2)=O)=O)CCN(C(=O)CC2CCC(F)(F)CO2)CC1 92901,N1(C(CCCCCC#C)=O)CC2CCCC(NC(C3CCNC3=O)=O)C2C1 92902,c1(CC(=O)NC2CC2NC(c2cc3scnc3[nH]2)=O)cccc(F)c1Cl 92903,c1(-c2cn(C(CNC(COCc3cc(C)no3)=O)C)nn2)ccccc1S(C)=O 92904,c1(C(C(F)(F)F)NCC(c2n(C)cnc2)O)cccc(C(F)(F)F)c1 92905,c1(OC)c(N(C2CCCN(C(C3CC4CCC3O4)=O)C2)C)ncnc1Cl 92906,c1(NC2CCN(C(c3cc[nH]c3C3CCCC3)=O)C2)cc(O)nc(O)n1 92907,c1(-c2cn(CCC(C(C)C)NC(C(C(=O)OCC)CC)=O)nn2)ccc2c(c1)CCC2 92908,c1(NCC2N(C(=O)CCC3CCCC(O)C3)CCCC2)ncc([N+](=O)[O-])c(=N)[nH]1 92909,C(=O)(CCC(C)C#N)NCC1CC(NC(c2c(CC)nn(C)c2)=O)C1 92910,C1(C)(C(N(CC(CNC(C2CC(CC)(CC)C2)=O)C)C)=O)CCC(C)C1 92911,C(=O)(CCC(C)(C)NC(=O)C(C)CC#N)N(C1(C(=O)OC)CC1)C 92912,Cc1ccc(O)nc1CNC(=O)CC(C)(C)CNC(C1OCCC1C(C)C)=O 92913,C(C(CC(C)C)C(=O)NCC1COCC(=O)N1C)NC(C(CC)=CCCC)=O 92914,CC(C)C(C(=O)N(C)CC1CCN(C(c2ccncc2Cl)=O)C1)NC(N)=O 92915,Cc1cc(C)c(C(N2CCCC(NC(=O)CSC(F)(F)F)C2C)=O)cc1N 92916,c1(C(=O)NCC2CC(OC)CN2C(C2CC(SC)C2)=O)cc(Cl)cc([N+](=O)[O-])c1 92917,c1(CCCNC(C(=O)NCc2c(OC)cc(C)s2)=O)cc(C)cc(C)c1 92918,c1(OC)cc(N)c(F)cc1CNC1Sc2ccccc2O1.c12ccc(cc1)OC2 92919,C(=O)(C(C)(C(C)C)OC)N1CCC(CCC(C)(C)CNC(CC=C)=O)CC1 92920,c1(C(N2CCN(C(C(CC3CCC3)C(=O)OC)=O)CC2)=O)ccnc2ccsc12 92921,C1(NC(C(CC)CO)=O)CC2(CCN(C(C3C=C3C)=O)C2)C1 92922,C1(CNC(C(=Cc2cccs2)C)=O)CCN(C(C2CC2C2(C)COC2)=O)C12CC2 92923,c1(C(=O)NC(C2(O)CCN(C(Cc3nc(C)[nH]n3)=O)C2)C)cccc2cncn12 92924,C(=O)(C(C)(C)CS(C)(=O)=O)N1CCCC(C(C)NC(c2c(SC)cccc2)=O)C1 92925,c1(COC(C(C)CCC(C)(C)C)=O)ccnc2cc(Br)ccc12 92926,Cn1nc(C(F)(F)F)cc1C(N1CCC1CNC(=O)CC1CCCS1(=O)=O)=O 92927,CC1CN(C(C2(CO)CCOCC2)=O)CC(C)N(C(=O)Cc2csc(Cl)n2)C1 92928,c1(C(=O)NCC2C(NC(C3(C(N)=O)CCC3)=O)C2)cccc(F)c1F 92929,C=CCCCCC(=O)NC(C)C(C)NC(c1cc(C2CCCCC2)on1)=O 92930,c1(OC)ccccc1C1CC1C(=O)NCCC(C)(C)NC(C1C(Cl)(Cl)C12CC2)=O 92931,N1(C(C(CC)F)=O)CCN(C(C2CC(N(C)C)C2)=O)CC1c1cnn(C)c1 92932,c1(CNC2CCC(C)CN2C(=O)OC(C)(C)C)nnc2n1CCOC2 92933,Cc1cc(CNC(c2[nH]ccc2C2CC2)=O)oc1C(=O)NCCC(C)(C)O 92934,C1(C(C)C)N(C(C2(CO)CCN(C(c3ccc[n+]([O-])c3)=O)C2)=O)CC1(C)C 92935,N1(Cc2n(C)cnn2)CCCN(C(C2C3CN(C(=O)N(C)C)CC23)=O)CC1 92936,C(=O)(C(CC(C)(C)C)OC)NC1CC2(CC(NC(CN(C(=O)OC)C)=O)C2)C1 92937,C1(CC(C)C)CC(NC(=O)C(N2CC(c3ccccc3)C2(C)C)=O)CCO1 92938,C1(C(N(C2CCN(C(=O)CCc3ccco3)CC2)CC#C)=O)CC2(CCC2)CO1 92939,c1(SCC#C)cccc(C(=O)NC(C)CCCNC(=O)C(C)OCC(C)C)c1 92940,N1(C(C(c2ccc(F)cc2)(C)F)=O)CCC(C2(NC(=O)C(F)CC3CC3)CC2)C1 92941,CC1=CCN(C(c2cc(CNC(C3(N(C)C)CC(F)C3)=O)on2)=O)CC1 92942,c1(C(=O)NCC2(C(=O)NC3(CC)CCCCC3)CCCCO2)n[nH]c2c1CCC2 92943,c1(CC(=O)NCCCCNC(C2(SCC)CC2)=O)ncnc2sccc12 92944,Cc1cnc(F)c(CNC(=O)C(c2ccoc2)NC(=O)C2=CCCCC2)c1 92945,N1(C(CN(C2CCC2)C)=O)CCCCC12CN(C(C1(c3ccno3)CC1)=O)C2 92946,c1(NC)cnc(Cl)cc1C(=O)N(C)CC1(O)CN(C(C2CCCC(C)C2)=O)C1 92947,c1(SC)nc2nc(C)c(CC(=O)NC3COC4(CCN(C(C)=O)C4)C3)c(C)n2n1 92948,C1(C(=O)NC(C#C)CC2CCCC2)C2CC3C(C2NC(c2cc(CO)[nH]n2)=O)C13 92949,N1(C(C(C)OCC)=O)CCc2ccccc2C1CNC(=O)Cc1ccsc1Cl 92950,C1(NC(=O)C=CC2CC2)CN(C(C2CC2C2CC2)=O)CCC1(F)F 92951,c1(C2CN2)cccnc1.N1(C(=O)OC(C)(C)C)CC(NC(C2CCCO2)=O)C1 92952,Cc1cc(CC(N2CCC(NC(c3cc(-c4ccccc4)co3)=O)C2)=O)cs1 92953,N1(C(C2CCC(NC(C3CC(C)(F)C3)=O)C2)=O)CC(CO)C(CO)C1 92954,N1(C(COc2cc(C)cc(C)c2)=O)CCN(C(=O)C=Cc2cocn2)C(C)C1C 92955,C=CCCCCC(=O)N1CCCOC(CNC(=O)CC(C)(C)C#N)C1 92956,c1(C(=O)NCCc2ccncc2)cnc2c(-c3csc4ccccc34)cnn2c1 92957,N1(C(C2CC(SC)C2)=O)CCCC1(C(=O)NCC(CC1CC1)CO)C(C)C 92958,C1(O)(C(C)NC(C(C)=C(C)C)=O)CCN(C(=O)Cc2nn(C)cc2Br)C1 92959,C1(CN(C(COCCCC(C)C)=O)C)CN(C(C2CCCCS2)=O)CCO1 92960,Cc1nnc2cc(N3CCCC(NC(=O)C(C)c4cccs4)CC3)ncn12 92961,c1(OC)cncc(C(C(=O)NC2CC2)N(c2c(C)cccc2Cl)CC2CC2)c1C 92962,c1(C(N2CCCC23CCC3)C(=O)NC(C(=O)OC)C)ccc(F)c(C)c1Cl 92963,c1(C(=O)NCC2CC2CNC(c2nnc(O)s2)=O)cc(Br)c[nH]1 92964,CC1CCN(Cc2ccccc2)CC1NC(=O)C(=O)NCC1CC2CCC1O2 92965,c1(NCC2(CC)CCCCC2)nc(N(C)CC2CCCO2)cc(C)n1 92966,Cc1ccc(C(N2CC(CC(F)C(=O)NCC3(O)CCC3)C2)=O)[nH]1 92967,C1(CNC(C(=O)NC2C(OC)CCC2)=O)CC(O)C12CCC2 92968,C1(C2CCN(C)CC2)(C(=O)NC(CC)CNC(=O)CCC2CC2(F)F)CC1 92969,C(=O)(C1=C(Cl)CCCC1)NCC1C2CN(C(CCNC(=O)NC)=O)C1C2 92970,O=S(=O)(c1cccc(=NCc2cc(CO)ccn2)[nH]1)N1CC2CC2C1 92971,CC(C)CC(C)C(=O)NC1(C)CCN(C(c2ccc(N)c(N)c2)=O)C1 92972,c1(C(N2CC(c3cn(CC(=O)OC)nn3)OCC2)=O)c(Cl)cccc1[N+](=O)[O-] 92973,C(=O)(C(CC)C(=O)N(C(C)CNC(=O)CCOc1ccccc1CC)C)OCC 92974,Cc1cc(C(=O)NC2CN(C(c3cncnc3C(C)C)=O)CC2O)c(C)s1 92975,n1(CCC(=O)OCc2cccc(OC)n2)nc(C)c(C)c1C 92976,N1(C(C#CCNC(C2(C)CCCO2)=O)=O)CCCc2occc2C1 92977,N1(C(C2(CCC)CCNC2=O)=O)CCC(CNC(=O)C(CC)SC)(COC)CC1 92978,c1(C(C(=O)NCC2CN(C(C(c3ccc(F)cc3)OC)=O)C2)C)cccc(F)c1 92979,c1(C(N2CC(CNC(C3CCCCC3)=O)C(F)(F)C2)=O)c(Br)ccc(F)c1F 92980,N1(C(Cn2ncn(C)c2=O)=O)CCCC1C1CCCN1C(=O)OC(C)(C)C 92981,c1(C(=O)NCC2(NC(C(CC3CCCC3)OC)=O)CCC2)ccn(C(C)C)c1C 92982,C1(C(N(C2CN(C(CC3CC(=C)C3)=O)C2)C)=O)CN=C2N=CNN2C1 92983,C12(C(N3CC(C(C)NC(=O)CCCN(C)C)C3)=O)CCCCC1C2 92984,Cc1c(CNC(=O)C=CCC(C)(C)NC(=O)Cc2cccnc2O)nnn1C 92985,C1(NC(c2ccc(C(C)C)s2)=O)CCC(NC(=O)CCC2CCCCN2C)CC1 92986,N1(c2nccc(N3CCC(C)CC3)n2)CC(NC(C2C=CCCC2)=O)CCC1C 92987,N1(C(CC2(C)CCCO2)=O)CC2CCCC2(NC(c2cc(O)cs2)=O)C1 92988,N#Cc1cccnc1CS(=O)Cc1cc(C2CC2)n(CC(F)(F)F)n1 92989,c1(-c2ccc(CNC(N(C)C)=O)o2)ccc(-c2cc(CO)ccc2C)cc1F 92990,C1(CNC2CC2c2ccccc2)CCC(C(=O)NCc2ccncn2)CC1 92991,c1(OC)csc(C(c2nnnn2Cc2cccs2)NCCCF)c1OC 92992,C1(CCC)CN(C(c2ccsc2C#N)=O)CC1C(N1CC2CC1CS2)=O 92993,C1(C(=O)NCC(C)(C)NC(c2nnc(C)s2)=O)CCCC(F)(F)CC1 92994,C(=O)(C(C)(F)C(F)(F)F)NCC(C(C)C)NC(c1cc(N)ccn1)=O 92995,c1(C(N2C(CCCNC(C3(C)CC3(Cl)Cl)=O)CCC2)=O)ncc(F)cn1 92996,C1(CC)CN(C(C23CCC(F)(CC2)C3)=O)CCN1C(c1cnn(C(C)C)n1)=O 92997,c1(OC)cc(O)c(NC(c2ccnn2CC2(C)COC2)=O)cc1C 92998,C1(C(=O)NC(C=CC(=O)N(CC)CC2CCCO2)(C)C)CC2C=CC1O2 92999,c1(C(=O)NCC(C)(CO)NC(=O)CCCCCC#N)nc[nH]c2ncnc1-2 93000,c1(C(N2CC(O)CC(NC(CC=C)=O)C2)=O)ccc2c(N(C)CC)ncnc2c1 93001,c1(C(=O)NC(C(C)NC(c2n(CC)cnn2)=O)C(C)C)c2c(c[nH]c1=N)CCC2 93002,C1(NC(c2ccc(C(F)F)c(F)c2)c2n(CCCF)nnn2)Cc2cscc2C1 93003,N1(C(c2c(NCC)scn2)=O)CC(NC(=O)CCOc2cccnc2)C2CC12 93004,C=CCC(C(=O)NCCCNC(c1cnn(C)c1Br)=O)NC(C)=O 93005,C1(COCC)(CN(C(=O)NCC2CC(F)C2)C)CCOCC1 93006,C12(C(=O)NC(CC)CNC(=O)CNC(C3CCCC3)=O)CCCC1C2Br 93007,C1(C(=O)NCC(CC)NC(c2cnc(Cl)n2C)=O)(OCC)CCCCCC1 93008,C(CCCCC(=O)N1CCC(NC(c2cn(C)c(C)n2)=O)CC1C1CC1)SC 93009,N1(C(C(C)C(C)O)=O)CCC2(CC1)CC(NC(=O)Cn1ncccc1=O)C2 93010,c1(NC(C)CCCO)nccc2nsnc12.c12ccccc1OC2 93011,c1(OC)c(C(N2CC3CCC3(NC(=O)CC3CC4(CC4)CO3)C2)=O)c(C)nn1C 93012,C1(C(N(CCOC)CCNC(=O)CCCCSC)=O)CCCC(F)(F)CC1 93013,c1(C(N(CCN(C(CN2CC(C)C2)=O)C)C)=O)cc(=O)c(Br)c[nH]1 93014,C1(CNC(C(C)c2ccsc2)=O)COCCN1C(c1sccc1Br)=O 93015,C(=O)(CC1=CCOCC1)NCC(CC(C)C)(C)NC(=O)Cn1ncnn1 93016,CC1(NC(=O)CC(Cl)Cl)CN(C(C2CS(=O)C2)=O)C1 93017,c1(C(=O)NC(CN(C(C(CC)NC(C)=O)=O)C)C)cccc(OC(F)(F)F)c1 93018,N#Cc1ccc(C(=O)N(CCCNC(c2cccn(O)c2=O)=O)C2CC2)cc1 93019,Cn1ncc(S(N)(=O)=O)c1C(=O)NCC1C=CCN1C(c1ccncc1)=O 93020,N1(C(C=Cc2c(C)ccnc2)=O)CC2CCC1CC2NC(C1CC12CCOC2)=O 93021,C1(NCc2nc(C)[nH]n2)CCN(C(=O)COC2CCCC2)CC1 93022,c1(COC)ccc(C(N2CC(NC(C3(C4CCCCO4)CC3)=O)C(O)C2)=O)cc1 93023,Cc1ncc(C=CC(=O)NCC2(F)CC(NC(=O)C(C)C3CCC3)C2)c(O)n1 93024,N1(C(CC2C(=O)NCCC2)=O)Cc2occ(C(N3CCC3C3CCC3)=O)c2C1 93025,C12(OC)CC(c3ccccc3)CN(C3CCCN1N=CN=C3OC)C2 93026,C1(C(=O)NC2CN(C(c3c(CC)cc(Cl)cc3)=O)CC2C)CNc2ccnn2C1 93027,CCCCC(CC(=O)NC(C)CCF)NC(=O)CC1CC2CCC1O2 93028,C(=O)(C(C)(C)CCCNC(C1CCCN(C)C1)=O)NCc1ccc(CC)o1 93029,c1cc(-c2cnc3cccnn23)c2c(c1)CN(c1ncnn3cccc13)CC2 93030,Cc1c(C(N2CCC(CNC(=O)C(C3CCOCC3)C)CC2)=O)cccc1O 93031,CON1CCC(C(=O)NCC2CC3CN(C(C4CC(N(C)C)C4)=O)CC23)CC1 93032,C1(C(=O)NC2(CC=C)CN(C(=O)Cn3nc(C)cc3N)C2)CC(=O)N(CCC)C1 93033,c1(C(N2CC(OCC(=O)NCC3(C=C)CCOCC3)C2)=O)ccc2cnoc2c1 93034,c1(C(=O)NCC(CCNC(C2(OC)CCCOC2)=O)O)cnc(C(F)F)c(C)c1 93035,Cn1cnc2c1CN(C(=O)CCCCNC(=O)Cc1csnn1)CC2 93036,c1(CC)ccccc1OCCC(=O)N1CC(CNC(=O)C=Cc2csc(C)n2)C1 93037,N1(C(C(C(=C)Cl)(C)C)=O)CC2CC(NC(c3ccc4nnnn4c3)=O)CC2C1 93038,c1(CC(=O)NC2(C)CC(NC(CCSCC)=O)C2)ccc(F)cc1F 93039,C1(C#C)(C(=O)NCCOCCCC#C)CCN(C(C2CCC(=O)O2)=O)CC1 93040,c1(CNc2cc(NC(c3cccnc3)CC)ncn2)cccc(O)c1Cl 93041,C(c1cnn(C)c1)=CC(=O)NC(C(=O)NCC1CN(C(C)=O)C1)C1(C)CC1 93042,c1(CC)cccnc1C(=O)N(C(C)CNC(C)=O)C.c12cccc(c1)CS2 93043,CC(C)(C(=O)NCC=CCNC(C1CNC(=O)C1)=O)c1ncco1 93044,c1(CNC(c2c(C(C)C)n[nH]c2)=O)cccc(NC(=O)CCc2cnccn2)c1 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93080,C1(CNC(c2n(CC)cnn2)=O)CCN(C(=O)CC23CCCC2C3)C1(C)C 93081,c1(CC(N2CC(NC(C3CCC3)=O)C3C2C3)=O)cc(F)cc(Br)c1 93082,CCC(O)C(C)(C)C(=O)N1CCC(Cn2cc(CNC(=O)CCCN=[N+]=[N-])nn2)C1 93083,S(=O)(=O)(CC(=O)N1CCCC(NC(C2CCCC(OC(C)(C)C)C2)=O)C1)N(C)C 93084,CC1(C(N2CCC(CNC(C3(CF)CCOCC3)=O)C2)=O)CC=CCO1 93085,c1(CC(=O)NCC2CN(C(CN(C)C)=O)C2)csc(NC=O)n1 93086,Cc1ncc(Br)cc1C(N1CC(N(C(=O)CC2CCC(C)(C)C2)C)C1)=O 93087,c1(CNC2CC(C(N3CCN(CC#C)CC3)=O)C2)cccc2nc[nH]c12 93088,Cc1cc(N)cc(C(=O)N(CCCNC(=O)C(c2ccccc2F)C)C)c1F 93089,c1(C(C)C)cccc(C(N2CCCCC2CNC(=O)C(C)(C)c2cscn2)=O)c1 93090,C(CN=c1[nH]c(=NCC2CCCN(CCCO)C2)[nH]c2c1COC2)OCCO 93091,c1(C(N2CC(CNC(c3n(CC)ncn3)=O)C2)=O)cccc(OC(F)(F)CF)c1 93092,N1(C(C2CCCC2)=O)CCN(C(=O)C=CC2CCCCC2)C(c2ccncc2)C1 93093,c1(C(=O)NC2CN(C(C3(C#C)CCCC3)=O)CC2O)ccc(Cl)c(C)c1Cl 93094,N1(C(C(C)SCC)=O)CC(CNC(=O)Cc2ccc(C)c(OC)c2)C(F)(F)C1 93095,C1(C(=O)NC2C(CNC(=O)Cn3cnc([N+](=O)[O-])n3)C2)CCC2(CCCCC2)C1 93096,c1(OC)ccc(O)c(C(=O)NC2CC(CNC(C3CC3Br)=O)C2)c1 93097,c1(C(N2C(CNC(c3cc(C)[nH]c3C)=O)CCCC2)=O)c(C)cc(O)nc1C 93098,N1(C(c2c(C)noc2)=O)C2CCC1CN(C(=O)C(C)CC1CCCO1)C2 93099,O(NC(=O)CC(C)NC(C1CCCN(C(C)C)C1)=O)CCOC(C)C 93100,N1(C(C2ON=C(C)C2)=O)CCCN(C(c2nc(=N)cc[nH]2)=O)C(CO)C1 93101,C1(NC(c2csc(C)c2N)=O)CC2(C1)CC(NC(=O)C(C)(C)CN1CCCC1)C2 93102,C=C(C)C(CC(=O)N1CCCC(N(C(C)C(=O)N(C2CC2)C(C)C)C)C1)OCC 93103,c1(C(=O)NC(C(C)NC(=O)COc2ccc(O)cc2)C)c[nH]c2cc(Cl)ccc12 93104,CCC(CCOC)C(=O)N1CCOC(CCCNC(=O)C#CC(=O)N(C)C)C1 93105,c12nc(C)ccc1CN2C.c1(OC)cc(C(C)OC(C2CCCCC2)=O)sn1 93106,Nc1nonc1C(N1CC(OCC(=O)NC2(C3CCCO3)CC2)C1)=O 93107,N1(C(c2cc(C)cc(C)c2)=O)CCCC2(NC(c3ccnnc3C)=O)CC2C1 93108,CC1OCCN(C(C2CC3(CCO2)CC3)=O)C1C(=O)NCc1cc(O)cc(F)c1 93109,N1(C(CC(C=C)C)=O)CC2CCCN(C(=O)CNc3ncccn3)C2C1 93110,C1(NC(CC2C(C)(C)C2)=O)CC2(CCCN(C(c3c(Cl)csc3Cl)=O)C2)C1 93111,c1(C(N(C)C)=O)ccc(CN=C(NCC(F)F)NC2CCC3CCC23)cn1 93112,c1(C(=O)NC2CCCC(NC(C3CN(C)C3)=O)C2)ccn2ncnc2c1 93113,Cc1cccc2[nH]cc(C(N3CC(C)(NC(C4CCC(C5CC5)C4)=O)C3)=O)c12 93114,N1(C(C(CCC)NC(C)=O)=O)CCCC(F)(CNC(C2SCCCS2)=O)C1 93115,c1(CC)ccc(F)c(C(=O)NCC2COCCN(C(=O)CC(C)C(F)F)C2)c1F 93116,N1(C(C2C(C)(C)C2)=O)CCN2CCN(C(=O)CN3CCC(=O)CC3)CC2C1 93117,C1(CNC(CC2(C)OCCO2)=O)CC(C(F)(F)F)CCN1C(=O)CCCN=[N+]=[N-] 93118,C(=O)(C1=NN(C2CC2)C(=O)CC1)N1CCC(O)(CN(C(=O)Cc2ccon2)C)C1 93119,C(C(C(=O)NCc1nccn1CC)C(C)(C)C)NC(c1oc(CC)c(C)c1)=O 93120,N1(C(C=CCCC=C(C)C)=O)CCC(NC(c2ccc(Cl)cc2C)=O)C(CO)C1 93121,CC(C)(C(=O)N1CCC1NC(=O)CN1C(=O)NC(C2CC2)(C2CC2)C1=O)C(F)F 93122,C(=O)(C(C)CCCC(C)C)NC(CC=C)CNC(=O)C=CC(=O)N(C)C 93123,N1(C(=O)C2CC2)CCC(F)(c2cn(-c3cccc(Cl)c3Cl)nn2)CC1 93124,c1(NC(C2CCN(c3cc(OC)nc(OC)n3)CC2O)=O)ccc(C#N)nc1C 93125,N1(C(c2cnc(C)nc2C)=O)CCCC2(CCN2C(=O)C(c2ccccc2)O)C1 93126,CCC(O)C(C)(C)C(=O)NCCN(C(=O)CCN(C1CCCCCC1)C)CC 93127,c1(C(=O)NCC(CCNC(c2ccc(C#C)cc2)=O)O)c(C)cc(C)cc1C 93128,c1(OCC(=O)NC)cccc(CC(=O)NCC#CCNC(=O)CC=C(C)C)c1 93129,C1(CNC(C(C)C2CCCO2)=O)(CO)CCN(C(=O)C=CCN2CCCC2)CC1 93130,N1(C(CN(CCC)C)=O)CCCCC1CN(C)C(c1cnn(C(C)C)c1F)=O 93131,Cc1cccnc1C(=O)NCCN1CCCC1CC1CCCN1C1CCCC1 93132,c1(OC)cccc(C(O)C(=O)NCC2CC2NC(c2cccc(C(C)C)c2)=O)c1 93133,CCCCC(O)C(=O)N1CCCC1(C)CNC(=O)CCSc1n[nH]c(C)n1 93134,c1(C(N2CCC(C(C)(C)O)(CO)C2)=O)cc(F)cc(F)c1O 93135,N1(C(c2c(C)cc(C)o2)=O)CCC(NC(=O)C(C)CN2CCOCC2)C12CC2 93136,C1(NC(c2cc(CSCC)on2)=O)CN(C(=O)C(C(C)(C)C)SCC)CCC1(C)C 93137,c1(NC2(CNC(C(C=C)O)=O)CC2)cnc(C#N)c(C#N)n1 93138,S(=O)(=O)(c1ccc(C=CC(=O)NC2CCSC3(CCC3)C2)cc1)NC(C)(C)C 93139,C(=O)(CCCC(=O)NCC1CC(OC)CN1C(C1CC1(C)C(F)(F)F)=O)OC 93140,c1(CC)nn(C)cc1C(=O)NCC(n1cc(CC2CCCCC2)nn1)C 93141,Nc1cccc(C(=O)NCC2CCCCN2C(C2CCC2(F)F)=O)n1 93142,c1(C(N2C3CC(NC(C4CCS(=O)(=O)N4)=O)C2CC3)=O)ccc2nnnn2c1 93143,C1(CNC(NC(CC)C)=NCC2CC(SC)C2)C(F)(F)C12CCOCC2 93144,c1(C(=O)NCC2(COC)CN(C(C3CN(C)C3)=O)C2)cc(Cl)cnc1OC 93145,c1(OCCC)ccccc1F.C1(N2C(=O)C2)CCN(C(=O)CC(=O)N(C)C)CC1 93146,C1(NC(C2N(C(C(C(C)C)OCC)=O)CC(=O)C2)=O)CC(C)(OC)C1(C)C 93147,C(=O)(CCC(C)(F)F)N1CCC(CN2CCN(C(C3C(C)OCC3)=O)CC2)CC1 93148,c1(C(N(C2CCN(C(C3CC(n4cnnc4)C3)=O)C2)CC)=O)cc2cscc2s1 93149,c1(C(N2CCC(N3CCN(C)C(=O)C3)C2)=O)cc2ccc(Cl)cc2s1 93150,C1(C2CCCC2)(NC(C2C3CN(C(C(CCC)F)=O)CC32)=O)CCC1 93151,N1(C(C2C(C(=O)OC)C2)=O)CCC2(CCN(C(c3nc[nH]c4nccc3-4)=O)C2)C1 93152,c1(C(N2CCOCC(CNC(C(C)(O)C3CC3)=O)C2)=O)cccc2scnc12 93153,N1(C(C=CCC)=O)CCC2CCN(C(c3c(C)[nH]c4ccc(O)cc34)=O)CC2C1 93154,C12(C3CC3)CCN(CC1)C2.Cc1nn(Cc2ccccc2)cc1C(=O)N 93155,C(=O)(CC(C)(C)CNC(C1(C)CC(=O)C1)=O)NC(C(=O)N(CC)CC)C 93156,C1(NC(CCCCN(C)C)=O)CCN(c2ncnc3c2nnn3C)CC12CCC2 93157,CC1OC2(C)CC1(C(=O)NC1CCN(CCOCC(F)(F)F)CC1)C2 93158,c1(CCC(=O)N(CCC(C)NC(=O)C(C)(C)c2cc[nH]n2)C)nnc(S)nc1O 93159,n1(CC(=O)NC2C(C)CN(c3ncncc3Br)CC2)ncc2ncccc12 93160,Cc1ncc(N(C(=O)CCC2CCN2CC)C(=O)C=Cc2ccccc2)cc1Cl 93161,C(=O)(C(C)(C)Cc1ccccc1)NC1CC(N(C(=O)COCc2nccs2)C)C1 93162,Cc1ccc(C(=O)NCC(C)CNC(=O)CC2COC(=O)C2)nc1 93163,c1(NC(C2C(NC(=O)CCC(F)(F)F)C2)=O)cc(Cl)nn2ccnc12 93164,c1(SCC)cncc(C(N2CC(CCNC(c3cn(CC)nc3C)=O)C2)=O)n1 93165,C(=O)(CC1=CCN(C(=O)CN2CCCC2)CC1)NCCc1nccc(C)n1 93166,N1(C(CNC(c2c(C)ccs2)=O)=O)CC(CO)CC1C 93167,N1(C(c2c(C)cccc2C)=O)CC2CCC1C(CNC(C1CC(=O)N(C)C1)=O)C2 93168,C#Cc1ccccc1CNC(=O)C(=O)N(CC(c1ccc(Cl)c(Cl)c1)OC)C 93169,C=C=C(C)CC(=O)NC1CC2(C1)CC2C(=O)NC1(CC=C)CCCCC1 93170,C(=O)(CC(CC(C)C)NC(=O)OC(C)(C)C)N1CC(CNC(C(C=CC)O)=O)C1 93171,c1(OC(C(N2C(C(C)NC(C(C)(C)OCC)=O)CCC2)=O)C)ccc(Cl)cc1 93172,c1(C(=O)NC2(COC)CCN(C(C3(C)CC3)=O)C2)ccc2c(c1)COC2(C)C 93173,c1(C(=O)NCCc2cccnc2)cnc2nc(NC(c3ncon3)=O)ccc2c1 93174,CC1CCc2ncc(C(N3CC4CCC3CN4C(=O)C(C)C(C)(F)F)=O)n2C1 93175,C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)NC(CC)CNC(=O)CCOC(C)C 93176,N1(C(Cc2c(C)cnn2C)=O)CCCN(C(c2ccc(OC(F)F)cc2)=O)CC1 93177,C1(=O)NNC(=O)CN1.c1(NC2N(C(C)C)CCC2)ccccc1Cl 93178,c1(OC)nccc(C(N2CC3(C2)CN(C(C2CCCCNC2=O)=O)C3)=O)c1F 93179,CCC(CC)(CC)C(=O)NCC1(F)CCN(C(=O)CC2CCCC(=O)N2)CC1 93180,c1(C(c2n(CC)nnn2)NCC(C2CCC(C(N)=O)C2)=O)ccc(C#N)cc1F 93181,c1(C(C(=O)NC2CCCN(C(C3(CC(F)F)CC3)=O)C2)O)cccc([N+](=O)[O-])c1 93182,C1(C(N2C(CCNC(C3(C#N)CC3)=O)CCCC2)=O)CCc2[nH]nc(O)c2C1 93183,CCC(F)(F)CC(=O)N1CC(CO)(NC(C2CC2(C)c2cccs2)=O)C1 93184,C1(NC(C(N2CCCCCC2)C)=O)CC2CCC1N(C(=O)CCC(N)=O)C2 93185,C#CC1CCCN(C(c2c(C(N)=O)cnn2C)=O)C1 93186,c1(C(n2c(C)cc(C)n2)OC)cc(C)c(C)nn1.N12CCCCC1c1cn(nn1)CC2=O 93187,C(c1cccc(O)c1)=CC(=O)NC(CNC(C1N(CCC)CCC1)=O)C(C)C 93188,c1(CC)ncncc1C(=O)NCc1cccc(-c2cccc(N(C)C)c2)c1 93189,CC1OC2CCC1(C(=O)N(CCCN(C(=O)COCC1(F)CC1)C)C)C2 93190,N1(C(C(N)=O)=O)CC(c2ccccc2)(NC(C2CC2F)=O)C1 93191,N1(C(c2cn(C)c(Br)c2)=O)CC2CC(CNC(=O)C=C3CCOCC3)C2C1 93192,c1(N2CC3N(C(C4(F)CCCC=C4F)=O)C3C2)ncnc2ccc(F)cc12 93193,C(=O)(C(=O)CC(C)CC)N(C(CNC(C(CCCC)O)=O)CC)C 93194,N1(C(c2c(CC)n(C)nc2)=O)CCC2CCN(C(c3cscc3SC)=O)CC12 93195,N1(CC)CCOC(C(=O)NC(C)C=CC(=O)NOCCNC(C)=O)C1 93196,N1(C(c2cn(C3(C(N)=O)CC3)nn2)C(=O)NC2(C)CC2)CCN(CCCF)CC1 93197,c1(N2CCN(C(C(CCN(C)C)(C)O)=O)CC2)ncc([N+](=O)[O-])cc1Br 93198,S(=O)(=O)(c1ccc(C(N2CCC(NC(=O)CC34CCCC3C4)C(O)C2)=O)o1)NC 93199,N1(C(C2CCN(C)CC2)=O)CCC(O)C(C(=O)N(C)Cc2cc(F)ccc2F)C1 93200,C(=O)(C(CN(C)C)CC)NC1C=CC(CC(=O)NCCCSCC)C1 93201,CC(C)(Cc1nn[nH]n1)C(=O)N1CCOCC1C(=O)NC1CCCCC1 93202,C1(NC(C(F)=CC)=O)CC(CNC(c2ocnc2C)=O)C1(C)C 93203,CC1(O)CCCN(C(=O)C(CC2CCC2)NC(=O)CCN2CCCC2=O)C1 93204,C1(C(NOCCOCC)=O)CN(C(=O)C=CC(F)F)CC12CCC2 93205,N1(C(CC2CC(C)C2)=O)CCCN(C(c2ncc(F)cc2F)=O)CC1C 93206,C1(C(=O)NC(C(C)C)CCO)CC(C)(C)CCN1C(=O)C=CC(F)F 93207,c1(NCCCNC(=O)NC)ccc(S(=O)(=O)NC(C)CS(C)=O)cc1Cl 93208,c1(OC)cnnc(C(=O)NCC(C2CC2)NC(C2(OC)CCOC2)=O)c1 93209,C1(C(N2CC(C)(NC(C3N4CC(C)N(CC4)C3)=O)C2)=O)CCc2nnc(O)n2C1 93210,c1(C(=O)NCC(C(C)C)NC(C2CC3(C2)CC3(F)F)=O)cccc(C(N)=O)c1N 93211,c1(C(N2CC(=CCNC(C(=Cc3ccccc3)CC)=O)C2)=O)cc(C)cc(Cl)n1 93212,C1(COC)CCN(C(=NCc2ccc(C3(C)OCCO3)cc2)NCC(F)F)C1 93213,C1(F)(CNC(C(C)Cn2cccn2)=O)CCN(C(=O)CN2CCCNC2=O)C1 93214,c1(C(C(=O)NCCCC2N(C(C(C3CC3)SC)=O)CCC2)F)cccc(F)c1 93215,C1(N(C)C(C2(NC(=O)C(C3CCOCC3)F)CSC2)=O)CCCCC1O 93216,c1(C(N2CCN(CCOC)C(C)C2)C(=O)NCC)cccc2sccc12 93217,c1(C(=O)N(C2CC2)CC2C(NC(c3c(CC)oc(C)c3)=O)C2)cnc(OC)c(Cl)c1 93218,C1(CCNC(CC=CC)=O)CC(F)(F)CN1C(=O)C(C)Oc1ccncc1 93219,C(C(N=c1nc(OC)[nH]c(OC)n1)C(C)C)NC(c1cc(CC)nc(Cl)c1)=O 93220,c1(CC)cnc(O)c(C(N2CCC(O)C(NC(C3SCC=C3C)=O)C2)=O)c1 93221,C(=O)(CC(C)(C)C#N)N(C(C)CC(=O)NCc1cn(CCNC(N)=O)nn1)C 93222,C1(c2noc(C)n2)(NC(C)C(=O)NC(c2cccc(F)c2)=O)CCN(C(C)=O)C1 93223,c1(C(=O)NCCN(C(=O)C(F)CC2CCC2)CCOC)n[nH]c2c1CCCC2 93224,C1(O)(C(CC)C(=O)NC(CNC(C2CC2F)=O)Cc2ccccc2)CCCCC1 93225,C1(CNC(C2C(C)CC=CC2)=O)CC(C)(C)CN1C(=O)CCCSC(C)(C)C 93226,c1(CC(=O)NCCOC2CN(C(=O)Cn3nnnc3C3CC3)C2)ncc(Cl)s1 93227,C(=O)(CC(O)CCSC)NCC(CN(C(c1scnc1C1CC1)=O)CC)(C)C 93228,C1(OCC#C)CCCN(C(=O)Cc2nc(-c3ccc(F)cc3)oc2C)C1 93229,CC1(C)CC(O)C(O)CN(C(=O)NC2(c3cc[nH]n3)CC2)C1 93230,CC1CCC(NC(C2CC23CCSCC3)=O)CN1C(=O)CCN1CCCCC1 93231,c1(C(=O)NCc2scc(CNC(c3cccc(CC)c3)=O)n2)cc(Cl)ncc1O 93232,c1(C(=O)NCCN2CCN(C(=O)COC3CCOC3)CC2)cnc2sccn12 93233,C1(NC(=O)NC(CC)C(O)C(=O)OC(C)(C)C)CCCC1S(C)(=O)=O 93234,c1(CN(C)C(=O)NCCCO)csc2ccc(Br)cc12 93235,N1(C(C2C(C)(C)C2)=O)CCC(O)(C2(NC(c3cc(C(N)=O)ccn3)=O)CC2)CC1 93236,C1(C(=O)NCCCSCC)CCN(C(=O)CCCCCNC(N)=O)CCC1(F)F 93237,C1(C(=O)N(C)Cc2cnco2)(COC)C=CCN1C(=O)CN1CCCC1 93238,c1(N(C(CNC(c2cc(CCC)[nH]n2)=O)C)C)ncnc(Cl)c1Br 93239,CONc1cccc(C(N2CCC2(C)C2CCCCC2)=O)n1 93240,C=C(C)C1OCCCC1C(=O)NCC1C=CCN1C(c1ccnn1CC)=O 93241,C1(C(=O)NC(CC)CNC(c2snc(C)c2Br)=O)CC2(CCOCC2)C1 93242,Cc1nc2n(n1)CC(C(=O)N(C)CC1CCCN1C(=O)CCCC(C)C)CC2 93243,Cc1cnc(O)c(CNC(=O)CC(C)N(C)C(C2CCCOCC2)=O)c1 93244,C1(O)(CNC(CC(C)(C)N(C)C)=O)CCCN(C(c2nnn3c2CCC3)=O)C1 93245,c1(C(N2C(C)CC(NC(C=C(C)C)=O)C2)=O)ncnc2c1c(Br)cn2C 93246,N1(C(CCOc2ccc(C)c(Cl)c2)=O)CC2CCCN(C(C3CC3C)=O)C2C1 93247,C1(CC)CN(C(c2cc(C)co2)=O)CCC1NC(=O)C(CC)c1ccccc1 93248,N1(C(C2N(C(=O)OC(C)(C)C)C(C(=O)O)CC2)=O)CC2CCCC(O)C2C1.OCC 93249,C1(N(C(C23CC(CCC)(C2)C3)=O)CC)CCCN(C(C2(O)CCSCC2)=O)CC1 93250,N1(C(C2C(OC)CCC2)=O)CC(OC)CC1CNC(=O)CCCNC(=O)C1CC1 93251,C1(NC(=O)C=C2CCCC2)CCCCC12CCN(C(C1(CF)COC1)=O)CC2 93252,C(c1cc(F)c(O)c(F)c1)=CC(N1CC2C(N(C(COC(CC)C)=O)C)C2C1)=O 93253,C1(OC)CCCC(C(=O)NCC(C)(C)CN(C)C(C2CC(Cl)(Cl)C2)=O)C1 93254,N1(CC(C)NC(c2ccc[nH]2)=O)CCN(C(C2C=CCCC2)=O)CC1 93255,c1(C(=O)NCC#CCNC(c2cc(OC)no2)=O)cc(Br)c(C)nc1O 93256,c1(C(=O)NCC(C)(CC)NC(c2c(CC)cco2)=O)cc2oc(Br)cc2[nH]1 93257,c1(C(=O)NC(CC=C)CNC(c2[nH]ccc2COC)=O)cncnc1C 93258,N1(C(C(C=C)OC)=O)CCN(C(C2CC3CCCC3C2)=O)CC12CC2 93259,C=C1CCN(C(c2cc(CO)n(C)n2)=O)C(C(N2CCC(C)CC2)=O)C1 93260,Cc1cc(=NCCC=CBr)[nH]c(N2CCC(Cc3ccn(C)n3)C2)n1 93261,C1(NC(C2CC(=O)NC2)=O)CN(C(C2C=CCCC2)=O)C2(CCCCC2)C1 93262,C(=O)(C(O)C(C)(C)C)NC(CSCC)C(N1CCN(CC)C(C)C1)=O 93263,N1(C(C2CCN(C)C(=O)C2)=O)CCC2(CCCN2C(c2ccc(F)c(Cl)n2)=O)C1 93264,C1(CCNC(C2CCC(=O)O2)=O)CCN(C(=O)CC2CNC(=O)C2)CC1 93265,C1(SC)CCCC1N=c1cc[nH]cc1S(=O)(=O)NCc1csc(=N)[nH]1 93266,c1(CNC(C(CO)NC(CCCSC)=O)=O)ccc(C)nc1O 93267,C1(CN(C(C2C(C)C2)=O)C)CN(C(=O)C(CO)c2ccccc2)CCO1 93268,CC(CC(N)=O)C(=O)N1CCCCC(NC(c2cc(-c3ccc(Cl)s3)[nH]n2)=O)C1 93269,c1(OC)cc(C(=O)NC2CC(C(=O)NCCn3nncc3C)C2)on1 93270,c1(NC(C(N2C(C(CC)O)CCC2)=O)=O)cccc(-c2ccccc2O)c1 93271,C1(CN(C)C(C2CSCC(=O)N2)=O)CCCN(C(C2CC(=C3CC3)C2)=O)C1 93272,c1(OC)cc(N2CCCC(C(C)NC(=O)C(O)Cc3cnc[nH]3)C2)nc(C)n1 93273,CC(CCO)N=c1[nH]c2c(c(=NCC(CO)c3cccnc3)[nH]1)CCCCCC2 93274,C1(C(N(CC(O)CN(C)C(C2CN3CCC2CC3)=O)C)=O)CN(CP(C)(C)=O)C1 93275,c1(C(=O)OC)ccc(CCC(=O)NCCN(C(=O)CSC(F)F)C)cc1 93276,c1(C(C)(C)C)ncc(C=CC(N2CCCCC2CC(=O)OC(F)F)=O)s1 93277,Cc1c(F)ccc(C(N2CC3CC(CNC(C4CC(F)C4)=O)C3C2)=O)c1N 93278,C(=O)(C(C)CNC(=O)CCc1ccn(C)c1)NCC(=O)NC(C)C 93279,C1(C(=O)N)(C(n2cc(C(CCC)N(C)C)nn2)C)CCCCC1.C1CCCCC1 93280,C1(c2ccccc2)(C(=O)NC(C2CC3CCCC23)=O)CC2(CC2)C1.C12(CC1)CN2 93281,n1(CCC(=O)NC2CN(C(=O)CCCC(F)F)CCC2F)cnc([N+](=O)[O-])c1 93282,C1(NC(C2OCCN(C)C2=O)=O)COC2(C1)CN(C(=O)CN1CCC(O)CC1)C2 93283,C12(C(=O)NCC(=C)CCNC(=O)C=CBr)CCC(CC1)C(C)O2 93284,C1(C(=O)Nc2ccccc2NC)CCC(C2CCCO2)O1.Cc1ccccc1 93285,N1(C(C(C)OCCOCC)=O)CC(NC(C2CC2C(C)(C)C)=O)C(F)C1 93286,C1(CC)COC(C(F)(F)F)CN1C(c1ccc(C(F)F)cc1OC)C(=O)NC 93287,C1(C(=O)NCC(CNC(CCCC(C)(F)F)=O)O)CCS(=O)(=O)C12CCC2 93288,c1(C(=O)NCC2(C(=O)NC)CC2)cc(Nc2cc(CC3CC3)ncn2)ccn1 93289,C1(CNC(c2cc(CC)no2)=O)CCCCN1C(=O)Cc1ccccc1CC 93290,CN(C)C1CCc2cc(NC(c3ccc(F)cc3)c3nnnn3C(C)C)ccc21 93291,c1(C(N)=O)ccc(NCC(N2CCC(CCNC(c3cnc(Cl)s3)=O)C2)=O)nc1 93292,C1(O)(CCNC(CC2CN(C)C2)=O)CN(C(c2ncoc2Br)=O)C1 93293,c1(C(n2nc(-c3ccn(C)n3)nc2C(O)C(C)C)C)ccc(Cl)cc1 93294,C1(NC(C(C2CC(F)(F)C2)OC)=O)CC12CCN(C(c1cc(C(C)C)sn1)=O)C2 93295,C(=O)(C(C(C)C)n1cnnc1)N1CC(C(=O)NCCNC(c2cn(CC)nn2)=O)C1 93296,C1(C(N(C2CCN(C(=O)CN3CCOCC3=O)CC2)C)=O)CC(=O)N(C2CC2)C1 93297,C(=O)(C(C)(O)CCC)NCC(N(C(c1c(CCC)n(CCO)nc1)=O)C)C1CC1 93298,Cc1nc(C)n(CC(=O)NCC2CCCC2NC(c2nn(C)nc2C(F)(F)F)=O)n1 93299,c1(C(N2CCN(C(c3nnn4c3CSCC4)=O)CC2)=O)cccc2c1COC2 93300,Cc1cc(C)c2c(c1)CCC2NC(=O)N=S(C)(=O)C1CC(O)C1 93301,Cc1cn2cc(C(=O)NCC3CCN3CC(Cc3ccccc3)OC)nc2s1 93302,N1(CCC(c2cccc(CC)c2)=O)CCN(C)C(=O)C1 93303,c1(C2(C(N3CC(O)(CNC(=O)C(F)F)C3)=O)CC2)ccc(Br)cc1F 93304,Cc1cc(C(=O)NCC(O)CNC(=O)CNc2ccc(CO)cc2)cc(C)c1O 93305,c1(N(C2COCCOC2)C(=O)NCCC2CC(C)(C)C2)ccc2c(c1)CC2 93306,N1(C(CC2(COC)CC2)=O)CC2CCC1C1CN(C(C3CCC34CCC4)=O)CC21 93307,c1(CC)n[nH]c(CC)c1CC(=O)NC(C1CN(C(c2coc(O)n2)=O)CCO1)C 93308,c1(C(C)C(=O)OCC23CCCC(CO2)C3)c[nH]c2ccccc12 93309,c1(CC)ccccc1C(CNC(C1C2CC3C(C2)C13)=O)NC(c1csc(=N)[nH]1)=O 93310,CC1COCC(CNC(=O)CCCCN(C(=O)C=C2CCCCC2)C)O1 93311,CCCC(C(O)C(=O)N1CCC=C(C)C1)NC(=O)COC1CC1 93312,N1(CCc2cn(CC(=O)NC(CC)(CC)c3ncccn3)nn2)CC(O)CCC1=O 93313,Cc1ccccc1OCCC(=O)NCC(C)(C1CC1)NC(C12CCN(CC1)C2)=O 93314,c1(OC)c(C(=O)NCC(C)N(C)C(c2csc(C)c2C)=O)sc(Cl)c1Cl 93315,N1(C(CCCN(C(C)C)C)=O)C(C(=O)NC2(CC3CC3)CCC2)CCC12CC2 93316,c1(NC(c2nnnn2CCOC)(CSCCC)C)cc(C)cc(Br)c1C 93317,C1(CN(C(CC=C)=O)C)CCN(C(C2OCC2(C)C)=O)CC1 93318,CC1(C)CN(C(=O)CCSC2CCCC2)CC1CNC(C1(C)CNC(=O)C1)=O 93319,N1(C(C=CSC)=O)CCC(C2CCN(C(C3OCCO3)=O)CC2)C1 93320,c1(NC(c2cc(CNC(c3ccc(C=C)cc3)=O)sc2)=O)ccc(C#N)cc1O 93321,N1(C(C2N(C)CCC2)=O)CC2CC1CN(C(c1nccc3nn[nH]c13)=O)C2 93322,c1(C(=O)NCC2CCN(C(c3cc(CO)ccn3)=O)C2)cc2c[nH]nc2cc1Br 93323,CCCCC(C(=O)NCC1CCC(C(=O)N(CC(C)(C)O)C)C1)C(C)C 93324,S(=O)(=O)(c1ccc(Cl)c([N+](=O)[O-])c1)Nc1ccccc1.C12COCC1NC2=O 93325,Cc1c(C(=O)NC(C)CCNC(=O)C(C)(C)N(C)C)cnn1CC(C)(C)O 93326,c1(OC)ccc(NC(C2(CNC(=O)CC3CC4(CC4)C3)CCC2)=O)c(Br)n1 93327,N1(C(COC)=O)CC2COCC(C1)C2NC(=O)CCc1cncc(F)c1 93328,CCCCCCOC(C)C(=O)NC(C1(O)CN(C(C2CC(OC)C2)=O)C1)C 93329,c1(OCC)ccc2nc(N3CCC(N(C)C(c4cccc(Cl)n4)=O)C3)sc2c1 93330,C1(NC(Cc2cc(C)on2)=O)CN(C(c2sc(CC(C)C)nc2C)=O)CC1C 93331,Cc1cc(N2CCC(C)C(NC(c3ccc(C)s3)=O)C2)c(C#N)cn1 93332,C1(C(=O)NC)CCC(Cn2cc(C3CCC(C)(C)C3)nn2)CC1 93333,C1(C(=O)NCc2cc(C)c(NCC(C)C)cc2)CCc2nnc(O)n2C1 93334,C=C1c2ccccc2C(=O)N1CC(=O)NC1CC(C)N(C(c2cc(OC)n[nH]2)=O)C1 93335,Cc1cc2[nH]c(C(=O)N(C3CC3)CC3CCCN3C(=O)C=CI)cc2s1 93336,C1(C)(CNC(C=C(CC)C)=O)CCCN1C(=O)CC1CCOC1=O 93337,C(=O)(C1CCc2c(Cl)cccc21)N1C(CNC(C(C)S(N)(=O)=O)=O)CC(C)(C)C1 93338,C1(O)(C(=O)NCC2(NC(C3CC(=C)C3)=O)CC2)CC2CCC1C2 93339,C(=O)(C1COc2ccc(Cl)cc21)NC1(CCOC)CCN(c2cc(O)ncn2)C1 93340,C=CCC(C(=O)N1CCC(CCNC(=O)COCCCC(C)C)C1)C(C)C 93341,CC(C)P(=O)(CC(=O)N1CC(C)(NC(=O)CCCC(N)=O)C1)C(C)C 93342,C(=O)(C(O)CC(F)(F)F)NC(CC(C)NC(C(c1c(OC)cccc1)=O)=O)C 93343,N1(C(C(COC)N(C)C)=O)CC(NC(c2cc(OC)nc(C)c2)=O)CCC1C 93344,C(=O)(C(C)S(N)(=O)=O)NCC1C(C(=O)NCCCCC2C(C)C2)OCC1 93345,c1(C(N(C2CCN(C(=O)C(O)CC(C)C)C2)CCC)=O)cc2nc(F)ccc2o1 93346,c1(CC(=O)NCCN(C(=O)CC(C)OC)CC)cccc(OC(C)C)c1F 93347,N1(C(C(C)NC(CC)(C)C)=O)CCC=C(C(=O)Nc2n[nH]c3c2CCCC3)C1 93348,c1(N(C)CCOC(F)F)nc(N(C)CC2CN(C)C2)nc2ccc(Cl)cc12 93349,C=CC1OCCC1NC(=O)CC1CCN(C(=O)Cn2ccc(C)c2)CC1 93350,CCC(CC)CCC(=O)N1CC(OC)CC1(C)CNC(C1(c2ccsc2)CC1)=O 93351,O=C1CC2C(C(=O)NC3CC(C(=O)NCC4CC4[N+](=O)[O-])CC3O)C2C1 93352,CC(C)(C#N)CCC(=O)NC1CC(C)(NC(c2ccn3cccc3c2)=O)C1 93353,c1(C(=O)NCC(CNC(C(C(=C)C)(C)C)=O)C)ccc2c(O)nccc2n1 93354,C1(F)(CNC(C(C(C)OC)O)=O)CCC(CNC(c2cnc(Cl)s2)=O)CC1 93355,c1(C(=O)OC)cc(C(=O)NC2CC(N(C(=O)Cc3csc(C(C)C)n3)C)C2)no1 93356,c1cccc(C(N(CCC(N2CCC(NC(=O)CO)CC2)=O)CC)=O)c1.CO 93357,Cc1cnc(C(N2CCCC(C)C2CNC(=O)CNC(=O)C(C)(C)C)=O)cc1C 93358,O=C1CCC2(C(=O)OCC3OCCCO3)CCCC2C1 93359,c12ccccc1CC(=O)N2.C(=O)(C(C)CC1CC1)NC1CC(OC(C)C)C1 93360,C(=O)(C1=NOC2(CCC2)C1)NC1C(NC(c2ccc(C(N)=O)c(Cl)c2)=O)C1 93361,C12(CC)CCC(NC(=O)CC(C)SC)(CC1)CO2.C123CCC(CO1)(C2)C(=O)NC3 93362,c1(C(N2C(CNC(CC(C=C)CCC)=O)CC2)=O)cc2ccccc2nn1 93363,C1(NC(CSCCOC)=O)CCCN(C(=O)C(=O)NCC(F)(F)F)C1C 93364,c1(COC(Cc2cn(C(C)(C)C)nc2)=O)ccc(Br)c2cccnc12 93365,N1(C(CCN(CCC)C(C2COC(C)C2)=O)=O)CCOC(CN=[N+]=[N-])C1 93366,CC(C)CC(CN(C)C)N(C(=O)CS(N)(=O)=O)C(c1cnc(C2CC2)nc1)=O 93367,N1(C(C(CSC)(C)C)=O)CCC(F)(F)C(CNC(=O)CC2CC2(C)C)C1 93368,N1(C(CSCC)=O)CCCC12CCN(C(c1nccn3cnnc13)=O)CC2 93369,c1(OC)ncc(S(=O)(=O)NC(=O)Cc2cnn(-c3ccccc3)c2)cc1C 93370,N1(C(CC=CCC)=O)CCC(C)(C)C1CNC(=O)CC1CCC1C1CC1 93371,c1(C(=O)NC2C(CC(=O)NCC3(CC)CCOC3)C(O)C2)cc(Cl)cn1C 93372,CN(C)S(=O)(=O)NCC(N1CCC(O)(CCNC(=O)C=C2CCN(C)C2)C1)=O 93373,c1(C(=O)O)ccc(CNCC23CC2CN(C(c2ccc(Cl)cn2)=O)C3)c(Br)c1 93374,c1(CC)[nH]ccc1C(=O)NCCn1cc(C(=O)N(CC(O)CO)C)cn1 93375,C1(NC(=O)C=C2CCC2)CN(C(=O)CNc2ccccc2)CC2(CCOCC2)C1 93376,c1(OCC)cccc(C(=O)NCCOCCCNC(=O)Cn2cnnn2)c1N 93377,N1(C(C=CC2(C)COC2)=O)CCC2(CC2C(=O)NCCCn2ccnn2)C1 93378,C(=O)(C(Cn1cncn1)NC(c1ccn(C)n1)=O)NCCCOC(C)C 93379,N1(C(c2ccc(CN=[N+]=[N-])cc2)=O)CCC2(CC1)CC2NC(=O)C(N)=O 93380,C1(CNC(c2cc(COC)on2)=O)C(C)CCN1C(=O)CSc1c(C)n[nH]c1C 93381,Cc1cc(C#N)nc(=NCC(C)(C)NC(=O)CSCc2ccc(F)cc2)[nH]1 93382,C1(NC(COCC(=O)NC)=O)CN(C(=O)CCCn2cncn2)CCC1C 93383,CC(C(O)C(F)F)NC(c1ccc(CNC(=O)C=CC2CCCCC2)cc1)=O 93384,C(=O)(C(C)CC#N)NC(C(C)c1ccccc1)Cc1ccccc1 93385,C1(C2CN(C(=O)CC(C)O)C2)(NC(c2c(CC)n(CC(C)C)nc2)=O)CC1 93386,c1(N(C)C)nccc(NC(=O)NCC23CC(C(=O)OC(C)(C)C)C(C2)C3)n1 93387,C1(CC(=O)NC2CN(C(=O)CC3CS(=O)(=O)C3)C2)CCCNC1=O 93388,C1(C)(CC)CC(N=c2[nH]c(=NCc3nnc4n3CCOC4)[nH]c3c2CCC3)C1 93389,CS(=O)(=O)c1cccc(CN2CCCC(CNC(c3cccc(Cl)c3Cl)=O)C2)c1 93390,c1(OC)cccc(C(C)CC(=O)NCC2CN(C(c3nc(O)sc3C)=O)C2)c1 93391,c1(OC)c(Cl)ccc(C(=O)NC(CNC(=O)CCc2cnn[nH]2)C(C)(C)C)c1F 93392,C1(C(=O)NC2C(CNC(C(CC)=CC)=O)COC2)CCC(N(C)C)CC1 93393,N1(C(C2(C)CC3(CCC3)C2)=O)CC2(CCN(C(C3CCC4CC4CC3)=O)CC2)C1 93394,c1(C(C(=O)OC(C)C)(C)NC(=O)NC2C3CC4C(C3)C24)cccc(F)c1 93395,CCCC(C)CC(=O)NCCCOCCC(=O)NC(C)CC1CCC1 93396,Cc1cc(F)ncc1-c1cn(C2CCN(C(C3CCC3C)=O)CC2)nn1 93397,N1(c2nc(OC)c(Br)cn2)CC2(CCC2)CC1CNC(=O)Cc1coc(C)n1 93398,CCC(C)(C)C(=O)NC1CCOCC1NC(C1CC1C(F)(F)F)=O 93399,c1(CC)c(C(=O)NCC(CC(C)C)NC(=O)CC(=O)NCC2CC2)csc1C 93400,c1(C2CCN(C(=O)NC3CC(NS(C)(=O)=O)C3)C2)ccc(F)cc1F 93401,C1(C(CNC(C(F)OC)=O)(C)C)CCN(C(C2CCC(C(=O)OC)O2)=O)CC1 93402,C1(CC(N2C(C(N(CC(Cl)Cl)C)=O)C=CC2)=O)CC(O)C1(C)C 93403,O(N(CC)C(=O)C(CCNC(=O)CS(=O)CC)OC)CC 93404,C1(F)(CNC(C2ON=C(CC)C2)=O)CCN(C(C2CC3CCC3C2)=O)CC1 93405,c1(C(=O)NC(C)C(=O)N(C(C)CCO)C)ccc(=N)[nH]c1 93406,C1(Nc2ncc(CC)s2)CC(OC)C12CCN(C(=O)OC(C)(C)C)CC2 93407,c1(CNC(C2CCCN(C(N3CCCCC3)=O)CC2)=O)cc(Br)c(F)cc1F 93408,C1(CCNC(c2cn(CC=C)nn2)=O)CN(C(=O)C(F)=C(C)C)CC(C)O1 93409,C1(C)(C(=O)NC(c2ccccc2Br)C)CCN(C(=O)C(C)(C)O)C1 93410,C1(NC(c2cc(C)[nH]c2)=O)CC(C)N(C(=O)CCc2nnc(C3CC3)o2)C1 93411,c1(C(=O)NCCNC(C2C(C)OCCC2)=O)ccsc1S(N)(=O)=O 93412,C(=O)(N(OC)C1CCOCC1)C1CC(CNC(C)=O)OC1.C1(C(C)C)C(=O)N1 93413,C1(C)(CNC(COCC=C)=O)CCN(C(c2ccnc(C(F)(F)F)c2F)=O)CC1 93414,c1(C(C)(C)C)cccc(C(=O)NC2CC2NC(C2CCCN2S(C)(=O)=O)=O)c1N 93415,S(=O)(=O)(c1ccc(NC2CCCOC2)c(C#N)c1)NCC1(C)CC1(Cl)Cl 93416,N1(C(CCCC)=O)CC(NC(C2CCN(C)C2C)=O)C2(CC2)C1 93417,c1(CCC(=O)NC(C(C)NC(c2ccc(C)cc2)=O)C)c(Cl)cncc1Cl 93418,c1(C(=O)OCC)cc(C)c(C)c(Br)c1S(=O)(=O)N1CC(C(=O)O)C2(COC2)C1 93419,c1(C(=O)NCCC2(c3ccccc3)CCCO2)cc(F)cc2[nH]ncc12 93420,CCCC(CCC)CC(=O)NC1CC(=O)N(C2CN(C(=O)CC3CCOC3)C2)C1 93421,C1(C)(COC)CC(NC(C2CCC2)=O)CN1C(C1CCSCC1)=O 93422,C1(C(N2C(CN(C)C)CCC2)C(=O)NCC(F)F)CC2(C1)OCCO2 93423,CC(C(F)F)N(C(=O)CCN(C(=O)COc1ccsc1)CCO)C 93424,C1(NC(c2c(COC)nn[nH]2)=O)CC2CC(NC(=O)CC(C)CN(C)C)C2C1 93425,Cc1cc(C(N2CC(C(=O)Nc3cc(CO)cc(F)c3)C3(CC3)C2)=O)cnc1C 93426,C(=O)(C1CCCn2c(Br)cnc21)N(C)CCOCCN(C)C(C1COC1)=O 93427,C(=O)(Nn1cnn(CC)c1=O)C1(C)N(C(CC2CC(=C)C2)=O)CC(O)C1 93428,c1(OC)cccc(CN2CCCC(NC(=O)CC3CCC=CCC3)C2)c1O 93429,C1(C(N(C(C)CCNC(=O)COCCN(C)C)C)=O)CCOC2(CCCCC2)C1 93430,c1(C(=O)NC(C(c2ccc(OCC)cc2)O)C)cc(OC)cc2ccoc12 93431,CC1c2cc(Br)ccc2OC1CNC(=O)N(C1CC1)CC1CC1 93432,C(=O)(CC1CN(C)c2ccccc21)NC1(C)CN(C(C(CC(C)C)C)=O)C1 93433,CC1(C(N2CCC(F)(CNC(c3ccnnc3)=O)C2)=O)CCCCC1(F)F 93434,CCC(C)CC(C(=O)N(CC(C)(C)NC(=O)CSC)C)NC(=O)COCCF 93435,CN1CCCCCC1C(=O)NCC(O)CCNC(c1ccc(Cl)c(Cl)c1)=O 93436,c1(C(=O)NC(C2CCCN(C(c3nc(=N)cc[nH]3)=O)C2)C)[nH]nc([N+](=O)[O-])c1Cl 93437,N1(Cc2cccc(OCC)c2)CC(F)(F)CC1C#N 93438,c1(C(N2CCCN(C(c3ccc(=N)[nH]c3)=O)CC2)=O)n[nH]c2nccc(Cl)c12 93439,Cc1ncc(CCC(=O)N(C(CNC(C2CC2c2ccccc2)=O)C2CC2)C)o1 93440,N1(C(C(=Cc2ccco2)C)=O)CCN(C)C(C(=O)NCC2CCNC(=O)C2)C1 93441,C(=O)(C(C)CC(C)(C)C)NCc1c(C(C)NC(=O)CCN(C)CCO)cccc1 93442,N1(C(C(c2ccccc2Cl)(C)C)=O)CC2CN(C(c3csc(O)n3)=O)CC2C1 93443,c1(C(=O)NC(C(C)NC(C2=NOC(C)C2)=O)C)cccc2sccc12 93444,c1(CN2CCCC(O)(CNC(=O)C(=O)C3CC3)C2)c(Cl)cccc1[N+](=O)[O-] 93445,Cc1c(NC(C)C(C)C)cccc1C(N1CCC(NC(=O)C2=NOCC2)CC1)=O 93446,N1(C(c2nc(C)n(C)c2)=O)CC(NC(c2cn(C)cn2)=O)CC2(CCC2)C1 93447,N1(C(c2cc(CC)sn2)=O)CCN(C(c2cc(C)ccc2C)=O)C(C(C)C)C1 93448,C(=O)(C(CC(C)CC)NC(c1c[nH]nc1OC)=O)NCC(C(CC)C)CO 93449,N1(C(C(=O)NCCC(=O)NCCC)C)CCN(C(C2CCOC2)=O)CC1C 93450,c1(C(=O)OCC)ccc2[nH]cc(C(=O)NC(Cc3ccncc3)C(=O)NC)c2c1 93451,C(=O)(C(C)CC(=O)NC1CC2CC(NC(=O)Cc3cncnc3O)C1C2)OC 93452,C12(NC(CCSCC)=O)CCC(CNC(c3ccc(OC)s3)=O)(CC1)OC2 93453,c1(CNCc2c(C)c(Br)cnc2)cc2c(cn1)OCCO2 93454,C1(C(=O)NC(CC)CCO)CN(C(=O)C=CC2CC2)CC1OC 93455,O=C(C1=CCc2ccccc21)NC1CCN(C(C2C3COCC23)=O)C(C2CC2)C1 93456,C1(NC(C(CC2CC2)OC)=O)(CNC(=O)Cc2ccc(C(C)=O)s2)CCCCC1 93457,N1(C(C=CCCCC)=O)CC(NC(C23CCCC2C3)=O)CC12CCCCC2 93458,n1(CC)ccc(C(=O)N(C(C)CCNC(=O)CC2CCC(C)C2)C)cc1=O 93459,C1(C(=O)NCC2CCCN2C(=O)CC2(C(F)(F)F)CC2)CCCC2CCCCC12 93460,c1(OC)cc(Cl)c(C(=O)Nc2cccc(NC(C3C4COCC34)=O)c2)cn1 93461,c1(C(C)C)ccc2c(c1)CC(N=c1ccc3c(Cl)ccc(F)c3[nH]1)CCC2 93462,C(=O)(CC1=CCOCC1)NC1C2CCN(C(c3ccc(OC)cc3)=O)CC21 93463,N1(C(C(C)C2CC2)=O)CCOCC1c1ccc(C(=O)NC2CCCC(O)C2)n1C 93464,CC(C)C(O)C(C)C(=O)N(C)CC1CCCN1C(c1cccc(C(N)=O)c1F)=O 93465,C1(C(=O)NC2C(NC(CCCCOC)=O)CCCC2)CCC2(CCC2)CO1 93466,C1(C(=O)NC(C)CCNC(=O)C(F)=CC2CC2)CC12CCS(=O)(=O)CC2 93467,c1(CC)cc(C(N2CCCC2C(C)NC(c2sccc2COC)=O)=O)oc1CC 93468,C(=O)(C(C)(C)C(F)c1ccccc1)NCC1C(C)CN(C(=O)C#CC2CC2)C1 93469,Cc1nn(CCC(=O)N(C2CCCCC2NC(=O)C(F)(F)CO)C)c(C)c1C 93470,CC(C)S(=O)(=O)CC(=O)NC1CN(C(=O)CCc2cncc(O)c2)CCC1C 93471,C1(C(=O)OC)CN(N2CCOCC2C(C)(C)C)CCO1 93472,O=NN1CCCC1C(=O)NCC(CO)NC(c1csc(-c2cn[nH]c2)n1)=O 93473,c1(NC(C2CCOCC2)(CC)C)c(Br)cnc(F)c1F 93474,C1(Nc2cc(OC)nc(OC)n2)CC2CCCC(C1)N2C(=O)COCC(=O)OC 93475,CS(=O)(=O)c1ccsc1CN=c1ccnc(NC2CC(O)C2)[nH]1 93476,C=CCC(C)C(=O)NC(C)(CNC(c1cc(C2CCCCC2)[nH]n1)=O)CC 93477,c1(OC)ncnc(C(N2CC(OCCNC(C3CCCCNC3=O)=O)C2)=O)c1F 93478,C(=O)(CCCCC#N)NC(C(C)NC(c1ccccc1Br)=O)(C)C 93479,C1(N(C(C#C)=O)CC)CC(F)CN(C(=O)C(CC)N(C2CC2)CC)C1 93480,Oc1cccc2c1CN(c1nc(=NCC3CC4(C3)CC(O)C4)[nH]c3c1COC3)C2 93481,CCCC(C)(CCC)C(=O)NCC1CC(O)CN1C(C1CC2(COC(=O)N2)C1)=O 93482,C1(NC(C(CCC)NC(N)=O)=O)CC2CC1N(C(c1cnc(OC)c(C)c1)=O)C2 93483,c1(C(=O)OC)ccc(-c2nscc2O)cc1O 93484,C1(CNC(C2(C)C=CCCC2)=O)CCC2(CN(C(C3CCC(C)CC3)=O)C2)O1 93485,c1(C(N2CCC(O)(CNC(c3n(CC)nnc3)=O)C2)=O)c(Cl)ccc(Cl)c1Cl 93486,CCC(O)CC(=O)NC(C(=O)NCc1nc[nH]n1)c1ccoc1 93487,N1(C(c2c[nH]c(=NC)o2)=O)CCCC1C1CCCN1C(c1ccc(OC)cn1)=O 93488,C#CC(CC(C)C)NC(C1CCN(C(=O)CCc2csnn2)C1C(C)C)=O 93489,N1(C(c2cnc(CC)s2)=O)C2CCC1CN(C(c1cnnc(C)c1)=O)CC2 93490,CCC(O)C(C)C(=O)NC1CC(CNC(=O)CC(c2ccccc2)NC(N)=O)C1 93491,CC(C)C#CC(=O)N(C(C)(CNC(=O)COCP(C)(C)=O)Cn1cccn1)C1CCC1 93492,C1(C(=O)NCC(C(C)C)NC(C(C(=C)Cl)(C)C)=O)CCc2nccn2C1 93493,Cc1cc(C(=O)OCCOc2ccccc2)c(Br)c(Cl)c1 93494,c1(-c2cccc(C#N)c2)cccc2nc(C(=O)Nc3ncc(Cl)cc3Cl)cn12 93495,c1(N(C)C)ncccc1C(=O)NCCC1CC(NC(c2[nH]c(C)cc2C)=O)C1 93496,c1(C(N2C(C(C)C)C(NC(=O)C(C)CN(C)C)CC2)=O)cc(F)cc(F)c1O 93497,N1(C(c2c(C)cc(SC)o2)=O)CCC(C)N(c2nccnc2F)CC1 93498,Cc1cc(C(N2CCN(C(C3CCSC3)=O)C(CC(F)F)C2)=O)c(N)c(Cl)n1 93499,c1(CNC(=O)CCC=Cc2ccccc2)ccnc2ncnn12 93500,N#CC1(C(N2CCC2CNC(=O)CC2CCSCC2)=O)CC=CC1 93501,C(=O)(N=c1[nH]sc2ncccc12)C1CC(C)CN1C(c1coc2ccccc12)=O 93502,c1(CC)cc(C(=O)NCC2(C)CCC(NC(=O)CNC(C)=O)C2)c(Br)s1 93503,C1(CNC(CC(=O)OC)=O)CCC12CN(C(=O)C(C)NC(=O)Cn1cnnn1)C2 93504,N1(C(C(CN(C)C)(C)C)=O)CCOC2(C1)CN(C(c1noc3ccccc13)=O)C2 93505,C(C)(CO)(C(=O)N1CCC(F)(CNC(c2cnc(O)n2C)=O)C1)NC(C)=O 93506,CC1CN(C(c2ccc(OCCF)cc2)=O)CC1c1cn(Cc2cccs2)nn1 93507,c1(N(C)C)ccc(N(C)C(C2CCOCCN2)=O)cc1 93508,C1(C(=O)NC(COCC)C)C2CCN(C(=O)CN3CCCCCC3)CC12 93509,C1(CC=C)(C(=O)NCCN(C(=O)C(O)CC)C)CCCCC1 93510,c1(C(=O)NC(CNC(C2(CC#C)CCC2)=O)C2CC2)c[nH]nc1C1CC1 93511,c1(C(=O)NCC(CNC(C(C(C)O)N(C)C)=O)C(F)(F)F)ncc2n1CCCC2 93512,C1(c2nnnn2C2CC2)(CCC(F)F)CCCC(C)(C)C1 93513,Cc1oc(C(N2CCN(C(=O)CC3CC(=O)NC3=O)CC2)=O)cc1S(C)(=O)=O 93514,N#Cc1ccc(=NCC2CCC(NC(c3cnc(Cl)[nH]3)=O)C2)[nH]c1 93515,c1(C(=O)NC(CC(C)NC(c2ccc(CCC)cc2)=O)C)ccc(OC)cc1F 93516,C1(CC)CCCCC1C(=O)NCCOCC(=O)NCCCN1CCCC1C 93517,C1(N(C(COCCCCC)=O)C)CCCC(N(C)C(c2csc(C#N)c2)=O)C1 93518,Cc1nc(N2CC(C)(C)CC2CNC(C2(F)CCCC2)=O)c2c[nH]nc2n1 93519,c1(OC)cccc(C(CNC(c2sccc2C)=O)NC(=O)CCNC(C)=O)c1 93520,c1(-n2c(C(=O)NCC3N(C(C(COCC)C)=O)CC=C3)ccc2)ccc(F)cc1 93521,C(=O)(C(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)N(C(CCNC(C)=O)C)C 93522,CP(C)(=O)c1ccc(C(=O)NC23CCCC2CN(C(C2CCC2)=O)C3)cc1 93523,C1(C(N(CCOC)CCNC(=O)C=Cc2ccoc2)=O)CCCC(C)CC1 93524,c1(CC)ccnc(C(=O)NC(C2CCN(C(c3cnn(C)c3SC)=O)CC2)C)c1 93525,C12(NC(c3cc4ccccn4n3)=O)COCCC1CN(C(=O)Cc1cc[nH]n1)C2 93526,C1(CNC(c2n(CC(=C)C)nnn2)c2cnoc2)Cc2ccccc2C1 93527,C(=O)(CCS(=O)(=O)N(C)C)N1C(C(C)C)C(NC(C2(C3CCCO3)CC2)=O)CC1 93528,C1(C(N(C)Cc2nncn2C2CC2)=O)C=CCN(C(=O)CC2CC2)C1 93529,N1(C(CC(CC)C)=O)CC2(C1)C(NC(=O)Cc1ccc(C)cc1)CCS2(=O)=O 93530,CC(CC(=O)NCC1(C)CN(C(=O)C#CC2CCOC2)C1)C(C)(C)C 93531,c1(C(N2CC3C(CC(=O)NC(C)(C)C#N)(CC3)C2)=O)ccc2c(c1)COC2 93532,N1(C(C(CCC)C)=O)CC2CC1CC2CNc1ccc(C2(C(F)(F)F)N=N2)cc1 93533,CCCCC(O)CC(=O)N1CC2C(CC(=O)NC(c3ccccc3O)C)C2C1 93534,CN=c1[nH]cc(C(=O)NCC2(NC(=O)C(C)Oc3cccc(C)c3)CCC2)o1 93535,C1(C(=O)NC(CC(C)C)C)CC(C)(C)CN1C(c1cnc(Cl)n1C)=O 93536,N1(C(c2c3scc(C)c3ncn2)=O)CC(NC(=O)C=C(Cl)Cl)CC12CCOCC2 93537,C1(CNC(C(C)Nc2scc(C)n2)=O)CCCCN(C(=O)C(C)CC(C)C)C1 93538,CC(C)(F)CCC(=O)NCc1cc(C(=O)NCCc2ccon2)co1 93539,c1(CC)n[nH]c(CC)c1CC(N1CC(CN(C)C(C2CCCOC2C)=O)C1)=O 93540,C1(C#N)(C(N(C)CC2CC(F)CN2C(C2CC(C)(F)C2)=O)=O)CC2CCC1CC2 93541,O=C1CN(C(C2CC3(CC3)CN2C(c2cc[nH]c2)=O)=O)CCCN1 93542,CC1CN(C(=O)N(C2CC(=O)NC2=O)C2CC2)CC(C)N1C(N)=O.c12cnn(c1)CCSC2 93543,CC1(C(N2CCC2CNC(c2cccc(C(F)F)n2)=O)=O)COCCO1 93544,c1(SC)nccc(N2CC(CNC(=O)C(c3cnn(C)c3)O)CC2C)n1 93545,N1(C(c2cnc(C)n2C)=O)CC2(C(=O)NCCCC(C)CO)CC1CCO2 93546,N1(C(CCNc2c(C)cccc2)=O)CCC(NC(c2cscc2F)=O)C(C)C1 93547,N1(C(c2csc(-c3ccoc3)n2)=O)CC2CCC(C1CO)N2C(c1csnn1)=O 93548,C1(O)(CCNC(C=C(C)C)=O)CCN(C(=O)C(C)C(c2ccco2)=O)CC1 93549,CCCC(CCC)C(=O)NC(CC1CC1)C(=O)NCC(F)(F)CC1CC1 93550,c1(CC)ccc(C(=O)N(C2CCC(NC(c3cc4sccc4[nH]3)=O)C2)C)c(C)n1 93551,N1(C(C)=O)CSCC1C(=O)NC(C)CCCNC(C1(c2ccccc2)CCC1)=O 93552,N1(C(C(CN(C)C)NC(c2cc(CCC)[nH]n2)=O)=O)CC(C)OCC(C)(C)C1 93553,C1(C(=O)NCCC(C)SC)CCN(C(=O)CCC2(N(C)C)CCC2)O1 93554,C(c1cn[nH]c1)=C(C)C(=O)N(C(C)CN(C)C(c1cnc(C)o1)=O)C 93555,C(=O)(C1Cc2c(Cl)cccc21)N1CCCC(N(C(=O)CCCN2CCCC2)C)CC1 93556,C1(NC(c2c(C(C)C)cco2)=O)CCN(C(C2CSC2)=O)CC1CO 93557,N1(C(CP(C)(C)=O)=O)CCC2(CCC2)C(NC(=O)COc2cccnc2)C1 93558,C1(S(N)(=O)=O)(C(N2CCCC(NC(CNC(CC(C)(C)C)=O)=O)C2)=O)CCC1 93559,N1(C(c2ccc(CSC)o2)=O)CCCN(C(=O)C(C)C(C)(C)C)CC1 93560,CC1=C(C(=O)NCc2nc(CNC(c3oncc3C)=O)cs2)CCC1 93561,CC1(C)CN(CC(=O)OCC2(F)CCS(=O)(=O)C2)CC(CO)O1 93562,C1(CNC(c2cncc(-c3ccccc3)c2)=O)CCc2ccccc2N1 93563,N1(C(C(CC)O)=O)CCN(C(c2ccccc2Oc2ccccc2)=O)CC(O)C1 93564,CCC(CC)CCCC(=O)NCC1(COC)CN(C(=O)CCCc2cccs2)C1 93565,N1(C(c2nc(OC)oc2)=O)CCCC2CN(C(=O)CN(C)CCOC(C)=O)CC12 93566,C(C(CC(F)(F)F)NC(=O)C(F)(F)CC1CCCO1)NC(C(CN(C)C)O)=O 93567,C(=O)(CCCCCS(N)(=O)=O)N1CC(C)C(CN)C1.c1(N(C)C)ncnc(=N)[nH]1 93568,C=CC1(NC(c2cn(CC)cn2)=O)CCCCC1 93569,[N-]=[N+]=NCCCC(=O)NC(=O)CSC1CCC1.C12CC(C1)CNC2=O 93570,Cc1cc(C)nc(CN2CC(F)CC2CN=[N+]=[N-])n1 93571,C1(CNC(C2C(C)=CCS2)=O)CC2(CO1)CN(C(=O)C(c1cccnc1)O)C2 93572,C#Cc1cn(C)nc1C(N1CCC(CC(=O)NCc2ncc(C)cc2C)C1)=O 93573,C1(NC(C2C(C)OCC2)=O)CCCN(C(C2CCN(c3ncccn3)CC2)=O)C1 93574,c1(OC)cc(N)ccc1C(N1CC(NC(=O)Cc2cn(C)nc2Cl)C(SC)C1)=O 93575,C(=O)(CCCN(C)N=O)N1CC(C)C(NC(=O)CSc2cnn(C)c2)C1 93576,c1(NC(c2c(CC)n(C3CCCC3)nc2)=O)ccc(=O)n(-c2cccc(F)c2)c1 93577,C1(CNC(=O)Cc2ccccc2F)CCN(C(=O)CSc2nc[nH]n2)CC1(F)F 93578,c1(C(C(=O)NCCN(C(C2C(OC(C)=O)C2)=O)C)OC(C)C)ccccc1 93579,C1(CC=C)(NC(=O)C(O)Cc2ccco2)CCN(C(=O)Cc2ccc(Cl)cc2)C1 93580,CC(C)(O)CCC(=O)NCC1CN(C(=O)Cc2cnccn2)CC1C(F)(F)F 93581,c1(N(C)C)ccc(C(F)(F)F)c(CNC(=NCC2CCC2)NC2CSC(C)C2)n1 93582,C12(C(C)(C)C)CC(C(=O)NC3(CO)CN(C(C4COC(=O)O4)=O)C3)(C1)C2 93583,c1(C(C)C)ccc(CC(=O)N(CCCCN(C)C(c2cnn(C)c2)=O)C)cc1F 93584,C(=O)(C1=CCSC1)NCC(=O)NCC(c1ncc(Br)cn1)(C)C 93585,Cc1c(C(=O)N(C)CC2(NC(c3scnc3Cl)=O)CC2)oc2ccccc2c1=O 93586,C1(C(=O)NCC2(NC(C(C)=O)=O)CCCC2)CCCCC1C(=O)N(C)C 93587,O=S(=O)(c1ccc(Br)cc1N1CCC=C(F)C1)NCC(c1cccs1)O 93588,C=CC1(C)COCCN1C(c1ccc(OC(C)C)nc1)C(=O)NCc1ccco1 93589,N1(C(C=CC(C)NC(CC2(CC)CCC2)=O)=O)CCC(CC2CCC2)C1 93590,CCC(CCCC(=O)NC(C)CCC(C)(C)C)NC(c1n[nH]cc1C)=O 93591,c1(OCC(C)=O)nc(C(=O)NCC2C3CN(C(CN(C)C(C)C)=O)CC32)ncc1F 93592,CC1(C)CC1(C(=O)NCC1CC(=C2CC2)C1)NC(=O)C=CCO 93593,C1(SC)CN(C(C2CCSCC2)=O)CC1NC(=O)CC1CCCN1C 93594,c1(CNC(Cc2c(C)nc[nH]2)=O)ncc(C(N2CCC(C(C)O)C2)=O)cn1 93595,n1(C(C)C)ccc(CC(=O)NCC(C2CC2)NC(c2csnc2C2CC2)=O)n1 93596,C1(C(=O)NC(C2(O)CN(C(c3ccccc3Cl)=O)C2)C)CCCC(C)(C)O1 93597,C1(F)(C(=O)NC(CC#CC)CO)CCN(C(c2sccc2C#N)=O)CC1 93598,C1(C(=O)NCCOC2CCN(C(Cc3c(C)con3)=O)C2)CC(=O)NC1(C)C 93599,N1(C(C=CC=CC)=O)CCN(C(=O)C(n2nnnc2C(C)(C)C)C)C(C)C1 93600,c1(C(N2CC(C)OCC2C(=O)O)=O)cc(Br)cc(S(C)(=O)=O)c1 93601,c1(CC(=O)NCC2OCCN(C(CCSCC)=O)C2)ccc(C)cc1Cl 93602,c1(C(C)=O)ccc(C(=O)N(CC(C)CNC(=O)C(F)C(C)C)C)nn1 93603,c1(C(=O)NCC2C(NC(=O)CN3CCOCC3)C2)ccc2cccnc2c1 93604,c1(C(N(C)CCNC(=O)CCOC2CCOCC2)=O)cccc(C#CC2CC2)c1 93605,N1(C(C2CSCC(=O)N2)=O)CCN(C(=O)CC2CN3CCC2CC3)C(CCO)C1 93606,c1(C(C)NC(C)Cc2cccs2)cccc2c1CNC2 93607,C1(C)(NC(C(CC)=CCCC)=O)CCN(C(c2coc(C(=O)OCC)n2)=O)CC1 93608,Cc1cc(C)c(C(=O)N(C)CC2CCN(C(=O)CC(C)C3CC3)C2)c(S)n1 93609,C(N=c1[nH]c(=NCCC2CCCCO2)[nH]c2ccc(Cl)cc12)c1ccc(F)cc1 93610,N1(C(C(C)NC(N)=O)=O)CCC2CCCC12C(=O)NCC#CC(F)(F)F 93611,N1(C(C(CC)NC(C)=O)=O)CC2(CNC(=O)C(C)COC(C)=O)CC(F)(C1)C2 93612,CC(C)CS(=O)(=O)CCC(=O)N(CC(O)CNC(=O)C(C)Cc1ccncc1)C 93613,C1(OC)(CNC(c2cnc(O)o2)=O)CN(C(=O)CNC(N2CCCC2)=O)C1 93614,c1(C(=O)NCc2ccc(CNC(=O)C(F)F)cc2)cc2cc[nH]c2cc1Cl 93615,c1(C(=O)NC2C(CN(C(CN3CCC(OC)C3)=O)C)CCC2)c(C)nc(C)n1O 93616,C#CCCCC(C)C(=O)NC(C)CC1CN(C(=O)CCc2ccc(Cl)c(Cl)c2)C1 93617,C(=O)(C1=C(Cl)CCCC1)N(C(C)(C)CC(=O)NCC1CC12CCOC2)C 93618,C1(OC)CCCCC1NC(=O)CN(C(=O)C=Cc1cncn1C)C(C)C 93619,c1(C(N2C(CO)CC(NC(C3=C(C)CC3)=O)C2)=O)cccc2ncnn12 93620,S(=O)(=O)(C1CCC(C)(C)C1)NCCn1c(C)csc1=O 93621,n1(CC)nc(C(=O)NC2(C(N3CCC(C(=O)OC)CC3)=O)CCN(C)C2)cc1C 93622,N1(c2ccc(C(=O)OC)cn2)CCCCC(NC(=O)CC2CCOC(CF)C2)C1 93623,CC1(C(=O)NCC2(CF)CCC2)CCCN1c1cc(-n2ccnc2)ncn1 93624,C1(NC(CC(=O)NC)=O)CC2CCC(C1)N2C(=O)C(c1ccc(F)c(F)c1F)=O 93625,N1(C(C(C(C)(C)C)=O)=O)CCn2nc(CNC(C3CCSC3)=O)cc2C1 93626,CC(C)(CNC(=O)COC1CCCC1)CC(=O)NCCCc1cncnc1 93627,c1(C(=O)NCC2C(NC(c3cc(OC)ncc3)=O)C2)cc2cc(Cl)ccc2o1 93628,N1(C(c2ccc(CC)o2)=O)CCCC(C)(CNC(=O)C(F)(F)CC2CC2)C1 93629,C1(NC(CSc2cccc(C)c2)=O)CC(NC(=O)Cc2cnc(C)[nH]2)C12CCC2 93630,CC(CC(=O)c1ccc(Cl)cc1)C(=O)N(C)Cc1nc(CCCl)co1 93631,C(=O)(NNC(=O)N1CCSC1)c1c(C)ncs1 93632,Cc1csc2ncc(C(N3CCCC(C)C3CNC(C3CCNC3=O)=O)=O)n12 93633,N1(C(C(N2CCCC2C2CCCOC2)C)=O)CCC(NS(CC)(=O)=O)CC1 93634,C(=O)(C(O)CC(F)(F)F)NC1CC(NC(=O)CC(C(F)F)n2ccnc2)C1 93635,C=C(C)C(C)(C)C(=O)N1CCCC1CNC(c1csc(SC)n1)=O 93636,N1(C(C(C2CC2)OCC)=O)CC(NC(c2ccc(=O)oc2)=O)C(C)(C)C1 93637,C1(NC(c2c(C(C)C)ocn2)=O)CC2CN(C(c3cc(C(C)(C)C)on3)=O)CC12 93638,c1(C(=O)NC2C3CN(C(CCNC(=O)C=CCl)=O)CC32)csc2cncn12 93639,Cn1cc(I)c2c(NC(=O)COc3ccc(C(=O)O)cc3)ncnc12 93640,c1(OC)nc(Cl)ccc1C(=O)NCCC(C)NC(=O)C(C)(C)c1cnsc1 93641,C1(OC)CC(C)CN(C(=O)CC2CN(C(=O)C(CO)N(C)C)CCC2C)C1 93642,c1(-n2c(C)nnn2)cc(C(=O)Nc2ccc(N(C)C)nc2)ccc1Cl 93643,N1(C(C(C2CCC2)OCC)=O)CCC(F)C(NC(c2noc(C3CC3)c2C)=O)C1 93644,Cc1cn2c(C)c(C(=O)NCC3(CNC(C4OCC4(C)C)=O)CC3)nc2s1 93645,CC1CC(CCNC(=O)CCCCN2CCCC2)CCN1C(=O)CC#N 93646,C1(C(=O)NC(CC2CN(C(C(CCC)=CCC)=O)C2)C)CCc2n[nH]cc2C1C 93647,c1(C(N2C(C(=O)Nc3n(C)ncc3I)C=CC2)=O)cc2ccccc2[nH]1 93648,Cc1ncccc1C(N1CC(CNC(C2CCCN2C)=O)C(C(F)(F)F)C1)=O 93649,c1(NC(c2cc(Br)nn2C)C)ccc(C(=O)N(C)C)c(Cl)c1 93650,C(=O)(C1CCCn2ccnc21)NC1CC2(CN(C(CCC=CC)=O)C2)C1 93651,C12(CNC(C(COC)O)=O)CCC(NC(=O)CC(C)C)(CO1)C2 93652,C1(CC)OCCC1C(=O)NCC1(C(=O)NC2CC(OC(C)C)C2)CCC1 93653,CC(c1ccccc1C)=CC(=O)NC(C)CCCCNC(c1nc(=N)cc[nH]1)=O 93654,C(=O)(CCCCNC(c1cn[nH]c1)=O)NC(C)CCN(C)C 93655,C1(C(C(=O)OC(C)C)NC(=O)OC)CCOCC1.N1(CC)CCCC1 93656,c1(CC)sc(C(=O)NCC2CC(NC(C3(C)CNC(=O)C3)=O)C2)cc1Br 93657,c1(-c2cn(CCC)nc2)cnn2c1CN(C(c1ccc(O)c(C)c1)=O)CC2 93658,C=CCC(C(=O)NCCN(C(=O)C(C)(CC)C(N)=O)CCC)C(C)(C)C 93659,C(=O)(CC(C(=O)N1CCCC(NC(C2CCCCNC2=O)=O)C1)NC(C)=O)OC 93660,c1(NC2CCC(NC(=O)CC3(O)CCCC3)C2)nc(Cl)nc2ccc(Cl)cc12 93661,c1(C(=O)NCC(C)(O)CNC(C2CCCCN2N=O)=O)c(Cl)cncc1Cl 93662,C(N=c1ncc2ccccc2[nH]1)C1CC(NC(=O)COc2ccccc2F)C1 93663,c1(C(=O)NC(C(C)NC(CCCOCC)=O)CO)cnc2c(c1)NC(=O)CN2C 93664,CC1(C)CCN(C(c2csc(Cl)n2)=O)CC1NC(c1csc2ccccc12)=O 93665,C1(CC(=O)NCc2cn(CCNC(C3(CC)CCCC3)=O)nn2)CCC(=O)NC1 93666,c1(C(=O)NCC(CNC(C(c2cccc(C)c2)O)=O)F)cccc2nn[nH]c12 93667,C1(C2CN(C(=O)NCC3C(C)CC3)C2)OCC1(F)F 93668,Cc1noc(C)c1NC(=O)CC1CCCCC1NC(c1conc1C(C)C)=O 93669,c1(NCC)ccc2c(c1)CCN2.c1(C(C(C)C)N(C(=O)C=O)CC)ccccc1C 93670,N1(C(c2c(C)n[nH]c2)=O)CCN(C(=O)COC(F)(F)C(F)(F)F)CC12CCC2 93671,c1(OC)cc(OC)c(CN2CCC(C)(NC(c3nc(Cl)sc3Cl)=O)C2)c(Br)c1 93672,c1(C(N2CC(N(C(C(C)NC(N)=O)=O)C)C2)=O)cnc(O)cc1C(F)(F)F 93673,C1(NC(C(=C)F)=O)CCN(C(c2ccc(-c3ccccc3)cc2)=O)CC1F 93674,N1(C(c2nc(CCC)sc2)=O)CC(CNC(=O)C(C)(C)OC(C)C)OC(C)(C)C1 93675,c1(CCC(=O)NC(CNC(COCC(=O)OCC)=O)C(C)(C)C)nnc(S)nc1O 93676,c1(C(N2CCCC(CNC(CN(C(C)=O)C)=O)C2)=O)c(Br)ccc(N)c1F 93677,c1(C(=O)NCC2CCN(C(c3c(CC)nccn3)=O)C2)c(C)sc(C)c1C 93678,N1(C(c2ccn(CCC)n2)=O)CC2CCC1C(CNC(c1cnn(C)c1N)=O)C2 93679,C#Cc1cccc(C(=O)NC(C2CCN(C(=O)CSCC(F)(F)F)C2)C)c1 93680,N1(CC(=O)NC(C)CN(C(=O)C(O)Cc2ccccc2)C)Cc2ccccc2C1 93681,C1(CCNC(c2c(C)cccc2)=O)CCN(C(C2COCC(C)(C)O2)=O)C(C)C1 93682,N1(C(C2N(S(C)(=O)=O)CCC2)=O)CC2CC(C(=O)Nc3ccc(Cl)cc3)C1C2 93683,c1(OC)cccc(C(N2CCOCC2C(=O)NCc2ccc(Br)c(F)c2)=O)c1O 93684,C1(NC(C2CCS(=O)(=O)C2)=O)CCN(C(C2CC(Cl)(Cl)C2)=O)CC12CCC2 93685,Cc1noc2ncc(C(N3CCN(C(=O)CC(C)CF)C(CO)C3)=O)cc12 93686,c1(CN(C2CC(SC)C2)C)cccc(-c2cnn[nH]2)c1 93687,C1(C(=O)NC(CC)CNC(=O)Cn2cc(C(F)(F)F)cn2)CC2CCCCCC12 93688,C1(NC(c2n(CCCC)ncc2)=O)CN(C(=O)Cc2ccc(OC)cc2)C2CC12 93689,c1(C2(CNC(NNC(c3ccc(=N)[nH]n3)=O)=O)CC2)nccc2ccccc12 93690,C1(NC(C=CSC)=O)COC2(CNC(c3cnc(N)c(Br)c3)=O)CC1C2 93691,c1(-n2cc(C(=O)NCCOCCNC(C3CC4CC4C3)=O)nn2)cccc(Cl)c1 93692,N1(C(c2cccc(OCC)c2)=O)CC(NC(c2cnoc2)=O)CC12CCCOC2 93693,N1(C(C2(CNC(CC3CCN(C)C3=O)=O)CCCC2)=O)CC2(C1)CC1(CCC1)C2 93694,N1(C(C(CC)SC)=O)CCCCC(C2CN(C(c3ccc(O)c(Cl)n3)=O)C2)C1 93695,C(=O)(C1=CC2(CCOC2)C1)N(CC(N1CCOC(C2CC2)C1)=O)C(C)C 93696,c1(NC(=O)Cc2ccc(S(=O)(=O)F)cc2)ccc2c(=O)[nH]ccc2c1 93697,CCC(CC)(CCNC(=O)C1=C(C)OCC1)NC(=O)COC(C)(C)C(F)(F)F 93698,C12(C(=O)Nc3ccc(C#N)cc3)C3C4C1C1C2C3C41C(N1CCCC(CO)C1)=O 93699,C12(NC(c3n[nH]c(C)c3Cl)=O)CCCN(C(c3cccc(Cl)c3F)=O)CC1C2 93700,c1(CC(=O)N(C)CC2(O)CN(C(c3ccc(C)s3)=O)C2)cn2c(nc1=O)SCC2 93701,C12(C(=O)NCC3(CC)CCC3)CCCC1CN(C(=O)Nc1ccc(F)c(Cl)c1)C2 93702,C=C(C)C(CC(=O)NC1CCC1CNC(=O)Cc1cn2ccsc2n1)OCC 93703,c1(C(=O)NCC(CC(C)C)NC(=O)COCc2nc[nH]n2)nccc2n[nH]cc12 93704,CC1COC(C)(C)CN1C(C1CCCCC1CNC(=O)CCc1ccoc1)=O 93705,CC1(NC(=O)C(=O)NC(C2CC2)=O)CCN(C(C2CC2c2ccco2)=O)CC1 93706,C(=O)(CC(C)C(F)F)NC(c1cccc(C)c1)CNC(C1CCN(C)C1)=O 93707,c1(OC)cc(O)ncc1C(=O)N(C1CCCC(NC(c2nc(C)oc2C)=O)C1)C 93708,C(C1CCn2ccnc21)NC(=O)NCCn1ncc(CC)c1 93709,C1(NC(c2c(CC)cccn2)=O)C(CNc2ncccc2C#N)CCC12CCC2 93710,N1(C(Cn2ncc(CC)c2)=O)CCOC(CN(C(=O)C=Cc2ccccc2)C)C1 93711,n1(CCN(C(=O)C(C2CCNCC2)F)CCSC)cc(C)cn1 93712,C#Cc1ccc(CC(=O)NC2CCCN(C(=O)CCOC)CC2)cc1 93713,c1(C(=O)OCC)ccc2sc(C(=O)OCC(C)OC(C)(C)C)c(C)c2c1 93714,C1(CNC(CCCCOCC)=O)CN(C(C2CC2C(C)(C)C)=O)CC12CC2 93715,C1(NC(C2C(C(=O)OC)C=C2)=O)CC2CCCC(C1)N2C(=O)C(C)(C)CF 93716,C1(CNC(=O)CNC(c2cscn2)=O)CC2(CCN(C(=O)C=C3CCC3)C2)CO1 93717,CC(C)CC(O)CC(=O)N1CCC1C(N1CC(c2nc(=O)o[nH]2)C1)=O 93718,C(=O)(C1CCCc2nn[nH]c21)N(C)CC1CCCN1C(C1(O)CC1)=O 93719,N1(CCOC(C)=O)CCCC(C(=O)NC(C2CCOCC2)CC)CC1 93720,c1(C(N(CC(C)NC(C2(C)CC=CCC2)=O)C)=O)ccc2c(c1)n(C)c(=O)n2C 93721,CC(c1ccco1)=CC(=O)N(C)CC1CCCN1C(C1CCC(=O)C1)=O 93722,c1(CC)ccc(C(N2CC3C(CNC(c4[nH]cnc4C)=O)C3C2)=O)cc1F 93723,N1(C(C2N(C(c3ccc(C)nc3C)=O)CCCC2)=O)CCn2cnnc2C1C 93724,c1(C(=O)NCC2CCCC(NC(CN(C)CC)=O)C2)cccc(O)c1Br 93725,c1(NC(c2ncc(-c3ccc(NC(C)=O)c(F)c3)cn2)=O)cc(C)cc(C#N)c1 93726,c1(C(N2CCC(N(C(c3ccc(CC)[nH]3)=O)CC)C2)=O)cnc(O)n1CC 93727,C(N=C(NCC(C)(C)C)N1CCCC(O)(CO)C1)c1cccc(CC)c1 93728,CC1(C(=O)NCC2CCCN(C(=O)CCCCC3CC3)C2)CC(F)(F)C1 93729,CC(CC(=O)NC1CC2(C1)CC(C)(C)C2)C(C)(C)NC(=O)CCN=[N+]=[N-] 93730,CCCCCCC(=O)NCC(c1ccccc1)CNC(=O)CC(C)C(C)C 93731,N1(C(C(OC)OC)=O)CCC2(CCC(NC(c3cccc(F)c3Cl)=O)C2)CC1 93732,c1(C(N2C(CC)CN(C(=O)C(O)C3CC3)CC2)=O)ccc2nnnn2c1 93733,Cc1coc(C=CC(=O)NCC(CNC(=O)Cn2cccnc2=O)CO)n1 93734,N1(C(C(C)OCC)=O)C(C(N2CC(O)CC2CC)=O)C2CC(O)C1C2 93735,c1(C(=O)NCC2(NC(C(CC(C)C)C)=O)CCCCC2)ccc2ncsc2c1 93736,C1(CN(C(C(CC)OCC)=O)C)CN(C(=O)C(C)NC(N)=O)CCO1 93737,N1(CC(=O)NCC(CNC(C2(C)CC(F)C2)=O)CO)CC(=O)NC1=O 93738,CCC(C)C(O)CC(=O)N1CCCN(C(=O)CCC(=O)c2cccnc2)CC1 93739,C1(C(=O)NCC2(O)CC(NC(c3c(C)cnn3C)=O)C2)CCC(O)CN1C 93740,N1(C(C2CC(CC)C2)=O)CC2CC(C1)CN(C(=O)C(F)(F)C1(O)CCCC1)C2 93741,C1(CC(=O)NC2C(CNC(Cn3cc(C(C)=O)nn3)=O)C2)NC(=O)NC1=O 93742,c1(OC(C(N2CC(NC(CC(C)O)=O)(CO)C2)=O)C)ccc(Cl)c(Cl)c1 93743,c1(NC(C2CCN2C(c2cc(I)ccc2F)=O)=O)ncc([N+](=O)[O-])cc1Cl 93744,c1(NC(C)CNC(=O)C(C)Cc2cnc[nH]2)ccc2c(n1)CC(C)(C)CC2=O 93745,N1(C(Cn2nnc(C)n2)=O)CC(C(=O)NC(c2cn(C)nn2)(C)C)CCC1(C)C 93746,C1(CC(=O)NC(CCC2CC2)C(=O)NCC23CCC(CO2)C3)CCCC2CC12 93747,CC1(C)CC(CNC(C2(C)CCC(=O)N2)=O)CN(C(=O)CCCc2ccsc2)C1 93748,CC(C)(CC(=O)N1CCCCC1CNC(=O)C=C1CCCCC1)C1CC1 93749,C(C)(CN=[N+]=[N-])NC(C=CC(=O)NC(CN(C(C)C)CC)C)=O 93750,C1(n2c(-c3ccc(Cl)cc3C)nc(C)n2)CC2CCC1(C)C2(C)C 93751,C=CCC(CC)NC(=O)C(c1ccoc1)NC(=O)C(CSC)NC(C)=O 93752,C1(CNC(CC(=O)NC)=O)CC(F)(F)CN1C(c1oc(CC2CC2)nc1C)=O 93753,CCCCC(C(=O)NCC1SCCS1)NC(C1CCN1CC)=O 93754,Cc1ccc(F)cc1CC(N1CCN(C)CC1CNC(C1CCOC1)=O)=O 93755,c1(C(N2CC(CC(C)NC(C3(CO)CCCO3)=O)C2)=O)cc(O)c2ccoc2c1 93756,C(c1sc2ccccc2c1Cl)=CC(=O)NCC(CN(C(CCC=C)=O)C)O 93757,CCC(C)(C)C(C)NC(=O)C(C)CNC(=O)CN1CCOC1=O 93758,N1(C(CCc2nc(C)sc2)=O)C2CCC1C(NC(c1nc(Cl)sc1C)=O)C2 93759,C12(C(=O)NCC(CC=C)NC(=O)CCOc3ccc(Cl)cc3)CC1COC2(C)C 93760,N1(C(C(C)O)=O)CCC(C(F)F)(CNC(c2cc(-c3cccc(Cl)c3)on2)=O)C1 93761,N1(C(c2snc(C)c2Br)=O)CCN(C(=O)C(C)C2CC2)C(C)C1 93762,C12(NC(CCC=C=C)=O)CCN(C(=O)CCN3CCOCC3)CC1C2 93763,N1(C(=O)Nc2c(SC)cccc2)CC2(C1)CN(Cc1csc(C(C)C)n1)C2 93764,N#CCCCCCC(=O)N1CC2C(CNC(=O)C3=CC4CCCC34)C2C1 93765,N1(C(C=CC(=O)N(C)C)=O)CC(C(C(=O)NCCC2CC(F)C2)N(C)C)C1 93766,c1(N(CCCN(C(Cn2nnc(C)n2)=O)C)C)ncnc2cc(Br)ccc12 93767,C1(NC(c2cnn(C(CC)CC)c2C)=O)CCC12CN(C(=O)CCC(C)OC)C2 93768,C(=O)(N=c1ccc(C2CCCCC2)n[nH]1)NCC1OCC(C)(C)C1 93769,c1(C(=O)NCC(C)NC(CC(c2ccc(C)cc2)C)=O)ccc2oncc2c1 93770,CC1(C)CC(CNC(C2CCCCNC2=O)=O)CN1C(=O)Cn1nnc(=N)[nH]1 93771,N1(C(CCCCCC=C)=O)CCC2(CCN(C(=O)CC3CSCCO3)C2)C1 93772,C1(CNC(CC=CC=C)=O)COC(C)(C)CN1C(=O)C(c1cccc(Cl)c1)C 93773,N1(C(C(C=C)O)=O)CCC(NC(c2c(CC)ncnc2CC)=O)C(F)C1 93774,c1(C(N2CC(N(C(COCCC=C)=O)C)C(O)C2)=O)cc(C(F)F)cc(SC)c1 93775,CC(CC(C)(C)C)C(=O)NC(C)CCCCNC(C1CCCC(C)C1)=O 93776,Cc1ccc(C)c(OCC(=O)NC(c2nnnn2C2CC(F)(F)C2)C)c1 93777,c1(C(N2CC(CCNC(=O)CC(C)=C(C)C)(OC)C2)=O)cnn(C)c1C(F)F 93778,C(CCC(=O)NCC1(O)CN(C(c2nccs2)=O)C1)=C(C)C 93779,c1(CNC(C(C)C)CO)ccccc1-c1cccc(C(=O)NCCCN(C)C)c1 93780,N1(C(CCCCOC)=O)CC2CC(NC(c3cc(C)nc(N(C)C)n3)=O)C(C2)C1 93781,C#CCC(CC#C)C(=O)NCCCN(C)C(c1ccc(C)nc1N)=O 93782,c1(C(N2CCC(NC(CCCOCC=C)=O)C2C)=O)cc(C)n(CC)c1C 93783,c1(C(N2C3C(NC(C(CC)n4cncn4)=O)C(C3)C2)=O)cnc2ncnn2c1O 93784,C=C(CNC(C1CC1(Cl)Cl)=O)CCNC(C1(C)CC1(F)F)=O 93785,CC1(C)OCCOC1CC(N1CCN(C(c2[nH]ncc2C#N)=O)CC1)=O 93786,C(=O)(C(CC(C)(C)C)OC)N1CCC(N(C(=O)CN2CCCNC2=O)CC)C1 93787,C=Cn1nccc1C(N1CC(OCC(=O)NCCC(C)N(C)C2CC2)C1)=O 93788,C1(Cn2cc(C3CCN(C)C3)nn2)CC2CCCC2N1C(=O)COCCCF 93789,C1(C(=O)NCC(C)NC(C2CCS(=O)(=O)CC2)=O)CCc2nc(O)[nH]c2C1 93790,c1(OCC(=O)NC(C)CNC(=O)C(c2ccc(F)cc2)F)ccc(F)c(Br)c1 93791,C1CCCS(=O)(=O)C1.CCCC 93792,Cc1nc(C(=O)N(C)C)ccc1C(N1CCN(C(c2ccoc2)=O)C(C)C1)=O 93793,Cc1nc(C2CC2)ncc1C(=O)NC1CC1NC(C1CCO1)=O 93794,C(CCN=c1[nH]cncc1I)N.N1(C(=O)CCc2cnn[nH]2)CCCCC1 93795,C(C)(C)(CCCNC(=O)COc1cccc(F)c1)NC(c1ccc(SC)o1)=O 93796,CC(CCN(C)C)C(=O)NC1(CC(=O)NCc2cncc(F)c2)CCC1 93797,C1(C(N2CC3C(NC(C(CSC)C)=O)C3C2)=O)CN(C)CCN(C)C1 93798,C(CC(=O)N1CCN(C(=O)CNS(=O)(=O)CC)C(CO)C1)(C1=CCCC1)OCC 93799,c1(C(=O)NCC2C3CN(C(C(CC)(C)COC)=O)CC32)c(F)ccc(OC)c1F 93800,c1(NC(C2CC(F)(F)C2)C(=O)N(CC(=O)OCC)CCC)ccsc1CC 93801,Cc1cc(C2CCCN2C(=O)Nc2nc(C3CC3)oc2C)cc(Br)c1 93802,C(C(CCS(C)(=O)=O)OC)Nc1c(N(CC)CC)ccc(Br)c1 93803,c1(C(N2CC(CCOC)N(C(=O)Cc3cnoc3)CC2)=O)cc2c([nH]1)CCCC2 93804,N1(CC(C)NC(c2onc(CC)n2)C)CCN(C(=O)C(C)(C)CF)CC1 93805,N1(C(C2CCN(C(C3CCC(CC)CC3)=O)C2C)=O)CC2CC(C)C2C1 93806,CCCCCC(O)CNC(=O)CN(C(=O)C(C1CC1)OCC)C 93807,C1(CCC(=O)OC)CC(c2ccc(NC(C=COCC)=O)c(F)c2)=NO1 93808,N1(C(C2CCC(C)N2C(C2C3CC4C(C3)C24)=O)=O)CCc2nc[nH]c2C1 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93951,c1(C(N(C)CC2(O)CCN(C(c3nnc(C)s3)=O)CC2)=O)cc2ccccn2c1 93952,N#Cc1cc(C(N2CCN(C(C3(Cl)CC34CCOCC4)=O)CC2)=O)ccc1F 93953,c1(C(=O)NCCCC(C)NC(CC(C(C)C)O)=O)cc2c(Cl)ccnc2s1 93954,Nc1nccnc1C(N1CCC1CNC(c1c(Br)n[nH]c1Br)=O)=O 93955,N1(CC)CC(NC(=O)C(CO)NC(=O)C(C2CCCCC2)C)C(C)C1 93956,C1(NC(=O)Cn2cc(Cl)cn2)CCC2(CC1)CC2NC(C12CC3CC1C2C3O)=O 93957,N1(C(c2n(CC)nnc2)=O)CC2CCCC1C2CNC(c1cnc(Cl)s1)=O 93958,c12ccc(o1)S(=O)(=O)N2.N1(N(C)C(c2ccccc2)=O)CC(CO)CC1=O 93959,C1(NC(=O)NCc2ccc(O)cc2)CCN(N(C(CC(=O)OCC)=O)CC)CC1 93960,c1(C(N2C(C(NOCC=CC)=O)CCC2C2CC2)=O)cccc(O)c1F 93961,N1(C(CCCOC)=O)CC(OC)C(NC(=O)CCCc2nccs2)C1 93962,CCC(C(=O)NCC(N(CC)CC)C1CC1)N(C(=O)CCN(C)CCO)C 93963,C1(COC)CN(C(c2cc(C)n(C(C)C)c2)=O)CCN1C(C1CN(C)C(=O)N1)=O 93964,CC(CC(=O)NC1CCCN(C(=O)CCCC2CCCCC2)CC1)C(F)F 93965,c1(C(N2C(CNC(C(C)Cn3ccnc3)=O)CC2)=O)ccc2cc[nH]c2n1 93966,C=CCC(C(=O)NCC1CCC(NC(c2cc(C3CC3)sn2)=O)CC1)C(C)C 93967,C(=O)(C(CCN(C)C)NC(=O)CCOC)NCC(C1CCCC1)OC 93968,C1(C(C)(C)NC(=O)CCN2CCC2)CCN(C(c2ccc(OCCF)cn2)=O)CC1 93969,c1(NCc2c(C)cc(C)c(C)c2)nccc(=NC(C)C2CC2)[nH]1 93970,N1(C(c2cc(C)c(Br)nc2)=O)CCC(C)(C#N)CC1 93971,C(CCN=c1nc(N2CCOCC2)cc[nH]1)N(C(C(C(C)S(C)(=O)=O)C)=O)C 93972,C1(CC)CC(OC)CN(CC(c2cc(Cl)cc(Cl)c2)O)C1 93973,Cc1cc(CC(=O)NCC(CC(C)C)NC(c2sccc2C)=O)n(C)n1 93974,c1(C(=O)NCCN(C(C2CC(=O)N(O)C2)=O)CC)ccc2cn(C)nc2c1 93975,N1(C(c2c(CC)noc2)=O)CCCC(COC)(NC(=O)CC(CC)C2CC2)C1 93976,c1(C(N2CC(C)CC(NC(c3nc(C)oc3)=O)C2)=O)c(F)ccc(F)c1O 93977,c1(SC)cccc(C(=O)N(CCCCNC(c2occc2C2CC2)=O)C)c1 93978,N1(C(c2cc(OC)ns2)=O)CC2CCCN(C(=O)C(CC(C)C)C(C)C)C2C1 93979,c1(C(N2CCC(CNC(c3ccccc3NCCO)=O)C2)=O)ccc[n+]([O-])c1 93980,c1(C2(C(=O)NC3CN(C(CC4CN(C)C4)=O)C3)CC2)ccc(Cl)c(F)c1 93981,C(N=c1[nH]c(=NC(C)C(C)F)[nH]c2cccnc12)c1cc(OC)nn1C 93982,C1(Cn2cc(CC3CCN(C(c4cnsc4)=O)C3)nn2)CCCCNC1=O 93983,c1(CC(=O)NC(CN(C(=O)C=C(C)c2ccsc2)CC)C)cc[nH]c(=N)c1 93984,c1(OC)cc(CCNC(C2C3CCCC3CN2C)=O)cc(OC)c1OC 93985,Cc1ccc(C=CC(=O)N(CC(O)CNC(C2(C)CNC(=O)C2)=O)C)cc1Cl 93986,N1(C(C(CCSC)O)=O)CC(C2CC2)(C(=O)NC2CC(CO)C23CCC3)C1 93987,N1(C(c2ncc(C(C)C)s2)C(=O)NCCCCCC)Cc2ncsc2C1 93988,N1(C(COc2ccn(C)n2)=O)CCCCC1CNC(c1cnc(Cl)[nH]1)=O 93989,CC(CC(=O)NCCC(C)NC(=O)Cc1csc(-c2ncccn2)n1)C(C)(C)C 93990,C(=O)(CC(C)(C)C(=O)N1CC2CC(NC(c3coc(C)c3)=O)C1C2)OCC 93991,N=c1[nH]nc(CC(=O)NC2CCC(NC(=O)CCN3CCC(F)C3)C2)s1 93992,C1(NC(c2ccc(F)cn2)=O)(CNC(=O)C(O)Cc2ccccn2)CCOCC1 93993,C(CCCCCC=C)NC(C(CN(C(c1c(C#C)c[nH]n1)=O)C)C)=O 93994,N1(C(c2c(C)occ2C(F)(F)F)=O)CCOC2(C1)CN(c1ccc(C#N)cn1)C2 93995,C1(CC)CCN(C(=O)Nc2cccc(C3COC3)c2)C(CO)C1 93996,C(CS(=O)(=O)CC(=O)N1CCC(C(C)(C)NC(C2CCCC(F)(F)C2)=O)C1)OC 93997,C1(C(N2CCC(N(CCO)C(c3ccccn3)=O)CC2)=O)C2CCC(C2)S1(=O)=O 93998,CC1COc2c(C(N3CC4CCCCCCC34)=O)cccc21 93999,c1(OC)ccc(C(N2CCC(NC(C3CC34CC4)=O)C2(C)C)=O)cc1CC1CC1 94000,N1(C(c2nn(CC)nc2C)=O)CCC2CN(C(C3CC(n4ccnn4)C3)=O)CC12 94001,C(=O)(CS(C)(=O)=O)NCC1N(C(CN(C)C(C2CCC(F)(C(=O)O)C2)=O)=O)CCC1 94002,C1(C)(C(=O)NCC2(OC)CN(C(=O)C(c3cccc(C)c3)(C)C)C2)CCC(C)C1 94003,C12(C(=O)NCC3(NC(=O)CCc4cncs4)CCOCC3)CCCCC1C2(F)F 94004,C1(NC(CCn2ncc(C)c2)=O)CCN(C(=O)C(F)C(C)C)CC1(C)C 94005,Cc1nc(C(=O)N(C)C)ccc1C(N1CC(C2(NC(=O)C(C)N(C)C)CC2)C1)=O 94006,N1(C(c2c(C)ccc(C)n2)=O)CCC2(CCN(C(c3onc(C)c3C)=O)CC2)C1 94007,C1(C(N2CCC(N(C)C)(CC)C2)=O)CCC2(CC2)N1C(=O)C=C(C)C 94008,N1(C(C(C)n2cccc2)=O)CCCC(C(=O)NC2CCCC(O)C2)CC1 94009,C1(COC)(CNC(=O)C(C)(C)SC)CCCN1C(=O)C=Cc1cncs1 94010,Fc1ccc(F)c(-n2cc(NCc3cccc(F)c3F)cn2)c1 94011,c1(C(=O)OC)ncc(Br)cc1NC(C1CCN(C(C2CC(C)(C)C2)=O)C1)=O 94012,c1(C(=O)NC(C)CCNC(=O)C(C)c2cccs2)ccn2c1CSCC2 94013,c1(C(N2CCCC(CN(C)C(C3CC4(C3)CC4F)=O)C2)=O)c(F)cc(O)cc1F 94014,C1(S(=O)(=O)c2ccc(Cl)cc2)(C(=O)NOCC2CC3CC3C2)CC1 94015,c1(C(N(C2CN(C(c3ncccc3Cl)=O)CC2F)C)=O)scc2c1OCCO2 94016,C(=O)(C(C)(C)C(=O)N1CC(OCCC(N2CCC(N(C)C)C(C)C2)=O)C1)NC 94017,N1(C(C)=O)CCCCC1C1CCN(C(C23CC(c4ccccc4)C2C3)=O)CC1 94018,c1(C(=O)NCCCCCNC(=O)C=C2CC2)ccc2c(c1)nc(O)n2C1CC1 94019,c12cccc(c1)N2.c1(N(C)C(c2cc(I)nn2C)=O)ncccc1Br 94020,Cc1cc(C(=O)NC2CCCC(CNC(=O)Cc3ccnc(F)c3)C2)nc(C)n1 94021,c1(OC)ccc(NC(C2(CCNC(=O)CC3CSCCS3)CCC2)=O)cc1F 94022,c1(C(=O)N(CCC(=O)NC(C2CCCN(CC)C2)C)CC)ccc(C#N)c(Cl)c1 94023,CC1OCCOC1C(=O)NC1(c2ccccc2)CCN(C(=O)Cc2ccsc2)C1 94024,CCC(C(=O)NCC(C1CCCC1)NC(c1cn2ccnc2cn1)=O)C(F)(F)F 94025,C=Cn1nncc1C(=O)NCC(CCNC(c1ccsc1Cl)=O)OC 94026,c1(CC(=O)NC2(CCNC(C3(C(=O)NC)CC3)=O)CCC2)cccc(F)c1Cl 94027,C1(CNC(c2scc(OC)c2)=O)CN(C(C2CC(C#N)C2)=O)CCN1C 94028,c1(OC)ccc2c(c1)OC(C)(C)CN(C(C1CN(C)CCO1)=O)C2 94029,c1(N(C(c2cccc(C(C)(C)C)c2)C(=O)NCCCF)CC)ccc(F)cc1F 94030,c1(C(=O)NCC(CCNC(CN(C2CC2)CC)=O)O)cccn(C)c1=O 94031,c1(CN2CCCC(C(N3CCC(CN(C)C)CC3)=O)C2)ccc(I)cc1F 94032,C1(CC)CC(O)CCN1C(=O)CCOC1CN(C(=O)CC2CCOC2)C1 94033,N1(C(C2(CO)CC(C)(C)C2)=O)CCCC(F)(C(=O)N(C2CCOCC2)CCO)C1 94034,n1(CCCC(=O)N(C(c2ccccc2)CNC(=O)C2=CCC2)C)ccccc1=O 94035,C1(C(N2C(CNC(=O)C3=CCCS3)CC3(CC3)C2)=O)CCc2nncn2CC1 94036,c1(C(N2CCC(C(=O)OC)C2)=O)sc(NC(C2CCCCC2)=O)cc1C 94037,c1(C(N(CC(=O)NCC2CCSC2)CCOC)=O)cnn(C(C)C)c1 94038,CCS(=O)(=O)CC(=O)NC(CCC1CC1)C(=O)NC1(CSC)CC1 94039,N1(C(C(C)OCC2CC2)=O)CCC(CNC(c2cc(O)n(C)n2)=O)C(O)C1 94040,C1(CCCCCNC(CCC#C)=O)CCN(C(c2ncn(C)c2C)=O)CC1 94041,N1(C(COCc2cc(C)no2)=O)CC(CNC(=O)C=C2CCSCC2)CCC1C 94042,c1(SC)ccccc1CC(N1CCC(C(=O)NC(C2CCCC2(F)F)(C)C)C1)=O 94043,n1(C(CC)CCO)cnc2c(N(C3CCOCC3)CCF)ncnc12 94044,C12(C(=O)OC)CCCC1N(C(c1csc3ccccc13)C(=O)NCC(C)C)CC2 94045,C1(NC(C(F)=C(C)C)=O)CC1C1CCN(C(c2nccc3cccnc23)=O)CC1 94046,c1(CN(C)C)ccc(C(=O)NC2(C)CCN(c3nnc(C4CC4)o3)C2)cc1 94047,C1(C(=O)NC(CC)(C)C2CC2)CC12CCN(C(=O)C(O)CCC(C)C)CC2 94048,Cc1ccc(C(F)F)cc1C(=O)NC1CC(C)(NC(=O)CC2CC=CCC2)C1 94049,c1(C(N2CCC(C(C)C)C2)C(=O)NCCC)c(C)nn(-c2ccc(F)cc2)c1Cl 94050,S(=O)(=O)(c1cccs1)N1CCC(C(N2CCC2C(F)(F)F)=O)CC1 94051,C1(NC(C(COCC)n2cc(CC(=O)OC)nn2)=O)CCC2(CC1)COC2 94052,C1(CNC(CCC2CCC(C)O2)=O)CCC2(CN(c3ccnc(C#N)n3)C2)O1 94053,CC1CCN(C(C2(C)CCOC(C)C2)=O)CC1CNC(c1nccnc1Cl)=O 94054,C(C(C)CN=c1ccnc(NCc2nnc(COC)s2)[nH]1)OC 94055,C1(C)(C(N2CCC(NC(C3(COC)CC(=O)C3)=O)CC2)=O)CCN(C)C1=O 94056,CCC(CNC(C12CC(CC(F)F)(C1)C2)=O)(CC)NC(c1cn(CCO)nn1)=O 94057,c1(C(=O)OC)sccc1S(=O)(=O)Nc1cc(C(=O)O)cc(C(C)C)c1 94058,C1(NC(C=NOC)=O)(CNC(=O)C(C2CC2)OCO)CCCCC1 94059,CCC(C)(C#N)C(=O)N1CC(NC(c2oncc2C)=O)C(C)C1 94060,Cc1ncc(C(N2CCC(CCNC(=O)Cc3csc(C)c3)C2)=O)c(C)n1 94061,c1(CC(N2C(CNC(C(CC)C(C)C)=O)COCC2)=O)c[nH]c2cnc(Cl)cc12 94062,c1(SCC)cc(CC(N2CC(C(=O)OC)C2)=O)cs1 94063,c1(C(=O)NCC2(OC)CCN(C(=O)CC3CCCO3)C2)cnc2ncccn12 94064,C(=O)(C(CCC(N)=O)NC(c1cc(O)ccc1Br)=O)OC 94065,N1(C(c2ccc(COC)[nH]2)=O)CC(C)CCC1CNC(c1nccc(C)n1)=O 94066,C1(CNC(c2ccc(C(C)(C)C)s2)=O)CN(C(=O)C2CC2)CC1C(F)(F)F 94067,C1(NC(c2cc(CC)on2)=O)CC(CNC(c2cc(C)c(C)o2)=O)C1(C)C 94068,C(=O)(C(O)CCCNC(c1c(C)ccnc1O)=O)N1CC(CC)OCC1 94069,N1(C(c2c(CC)cc(N)cc2)=O)CCCC2(NC(c3ccc(OC)s3)=O)CC2C1 94070,c1(NC(C)=O)ccc(CC(=O)NCC2CCC(NC(c3ccsc3C)=O)C2)cc1 94071,C1(CCNC(C2CCN(C)C2)=O)CCN(C(C2(c3cccnc3Cl)CC2)=O)CC1 94072,CCCC(O)CNC(=O)C(=O)NCc1cn(C2CCCNC2)nn1 94073,C1(NC(C2(C)CC(F)C2)=O)CCCCC1NC(=O)CSc1ccccc1Cl 94074,C1(C(=O)NCCC(C)NC(C(C)Cc2cccc(F)c2)=O)CC(C(C)(C)C)=NO1 94075,c1(NC(c2c(CNC(C(C3CCC3)OCC)=O)ocn2)=O)ccc(O)c(C)c1 94076,N1(C(c2cc(OC)ncn2)=O)CCOC(C)(CNC(=O)Cc2cccnc2C)C1 94077,CN1CCC(N(C(c2cc(Br)cs2)C(=O)NC(C)(C)C)C)C1 94078,CC1(C)CC(NC(=O)CCS)CCN1.C(C)(C)C1CC1 94079,c1(CC)cc(N)ccc1C(=O)NCC1CCCCN1C(=O)CCc1cnc(O)[nH]1 94080,c1(NC(=O)NC(CSC)C(C)(C)C)cc2cccc(F)c2cn1 94081,S(=O)(=O)(c1ccc(NCC(O)CCO)cc1Br)NC(c1n(C)ncc1)CO 94082,c1(C(=O)OC)cnc(C)[nH]c1=NCC(C)NC(=O)C1CCCc2n[nH]cc21 94083,CCCC(CNC(=O)C(=O)C(C)(C)C)C(=O)N1CC(N2CCCC2=O)C1 94084,C1(NC(C2N(C(C)=O)CCOC2)=O)CC2(C1)CN(C(=O)C(=O)NC1CC1)C2 94085,C1(NC(C2CCS(=O)CC2)=O)CCCN(C(=O)CCC2CCCCC2)CC1 94086,N1(C(N(C(=O)OCC(=O)NC(C2(CO)CC2)C)C)=O)CC(CO)C1 94087,Cc1cc(F)c(C(N2CCCC2CN(C)C(C2CC=CC2)=O)=O)cc1F 94088,n1(CCC)cc(CNC(C2CN(C(c3ccc[nH]3)=O)CCO2)=O)c(C)n1 94089,c1(OC)ccc(NC(=O)C2CC2)cc1NC(=O)NCc1ccccc1C(C)C 94090,c1(OC)ccc(C(N2CC3CC2CN3C(=O)C(CSC)OC)=O)c(N)c1F 94091,N1(Cc2cc(COC)no2)CCC(=O)N(CCC(C(F)(F)F)OC)C1=O 94092,C1(NC(=O)C=Cc2cscn2)CC2CCC1(CNC(c1cc(Cl)c[nH]1)=O)C2 94093,c1(C(=O)NC(CNC(C2(COC)CCCO2)=O)C)ccc(Cl)c(N)c1 94094,N1(C(c2nc(CC)sc2)=O)C2CCC1C(NC(c1cnc(C(F)(F)F)nc1)=O)C2 94095,C(CCNC(=O)CSC)(C(N)=O)NC(COC(CC)CC)=O 94096,c1(SC)ncc(F)c(NC(CCCCC2CCN(C(=O)OC(C)(C)C)CC2)=O)n1 94097,Cc1oc(C#N)cc1C(N1CC(CC(F)C(N2CCCC(CCO)CC2)=O)C1)=O 94098,CC1CSc2ccc(Br)cc2C1NC(c1c(N)sc2ccccc12)=O 94099,c1(N(CCN(C(=O)OC)CC)C(c2ccc(Br)cn2)=O)cccc(CC(C)C)n1 94100,N(C(=NCc1ccccc1)NCC12CC(C(=O)OC)(C1)C2)Cc1cnc(CC)o1 94101,CC1CNc2c(C(N3CC4C(CNC(c5cc[nH]n5)=O)C4C3)=O)cccc2C1 94102,n1(C(C)C)nccc1C(=O)NC(C1CCCN1C(C1CCC1C)=O)C 94103,C(=O)(CN=c1cc[nH]cc1)NCC1CCN(C(c2c(CC)noc2)=O)C1(C)C 94104,c1(C(N2CC(CNC(C(CC=C)OC)=O)C(C)C2)=O)cc2ccccc2o1 94105,c1(C(=O)NC2CCC(NC(CSCC(=O)OC)=O)C2)csc2cccnc12 94106,C1(C(N2CC3C(CNC(c4c(C)ccs4)=O)(C3)C2)=O)C(O)C(=O)N(C)C1C 94107,CC(C)(O)CC(=O)NC1CC1NC(C1(c2ccc(O)nc2)CCC1)=O 94108,c1(CC)ccc(C(=O)NCC2CCCCCN2C(C2CCC(=O)C2)=O)cc1Cl 94109,Cc1snnc1C(N1CC(c2ccccc2)(NC(c2cc(CF)on2)=O)C1)=O 94110,C(=O)(CS(=O)(=O)c1ccccc1Cl)NC(CNC(C1N2CC(C)N(CC2)C1)=O)C 94111,CCC(CCC(=O)NCCCC(C)NC(=O)CNS(N)(=O)=O)OC 94112,N1(CCC(=O)OC(CN(C(C)=O)CC)OC)c2ccccc2Sc2ccccc21 94113,Cc1nc(O)[nH]c1C(=O)NCC(C)(O)CNC(=O)CN1CCOCC1 94114,C1(C(N2CC(COC)(NC(c3ccc(C#N)o3)=O)C2)=O)CCc2n[nH]c(C)c2C1 94115,Nc1ccc(C(=O)NC2CC(CCC(=O)NCC(F)Cl)C2)nc1F 94116,C1(CNC(CSCC=C)=O)CC2CCC1N(C(c1cc(C)nc(N(C)C)n1)=O)C2 94117,N1(C(C(CC)SC)=O)C2CCC1CC(N(C)C(c1ccc(O)nn1)=O)C2 94118,c1(COC(C2CCC(C(=O)OC(C)(C)C)C2)=O)ccc2c(c1)COC21CCCC1 94119,N1(C(Cc2cc(C)cc(F)c2)=O)CC(NC(c2cccc(C)n2)=O)C2CCCC12 94120,C1(NC(C2CCC(OC)C2)=O)C2CC(NC(=O)CC3NC(=O)NC3=O)CC12 94121,c1(C(=O)NC2(CNC(C(C(C)C)F)=O)CC(F)(F)C2)nccc2n[nH]cc12 94122,c1(C2(C(C)(C)O)CC2)cn(CC(N2CCC(N3CCC3)C2)=O)nn1 94123,N1(C(c2ccn(CCC)n2)=O)CC2CC1(C(=O)N(CC(C)CO)C)C2 94124,CCC(C)(C)C(=O)N1CCCC(CC(=O)NCCCNC(=O)OC)C1 94125,c1(C(=O)NC2CCCN(C(C(C)N(C(C)=O)C)=O)CC2)cc2ccc(F)cc2[nH]1 94126,CN1CC(C)(C(=O)NCC2CC(NC(c3cccc(OC(F)F)n3)=O)C2)CC1=O 94127,C1(CNC(C=C2CCC(C)C2)=O)CN(C(=O)CC2(C)CC(F)(F)C2)CC1O 94128,c1(SC)cccc(C(=O)NC(C)(C)CCCNC(=O)Cn2cnnn2)n1 94129,c1(NCCCc2ccc(C(=O)Nc3c(CC)nccn3)[nH]2)c(F)ccc(Cl)c1F 94130,c1(C(N2CC(c3cn(C)nc3)OCC2)=O)ccc(F)c(N)c1 94131,C(=O)(C(CC)N(C1CCCCC1)CC)OC1CC(n2cc(C3(O)CCC3)nn2)C1 94132,C1(C)(C(=O)NCCN2CC(OC)C2)CCN(C(=O)CN2CCCCC2=O)C1 94133,C(=O)(C(C)(O)C(C)c1ccccc1)N(C1(c2ccccc2F)CCCCC1)C(C)=O 94134,C(=O)(C(C)(C)C(=O)N1CC(CC(=O)N(CCCCl)Cc2cccc(F)c2C)C1)OC 94135,C#Cc1cccc(C(=O)NC2CCOCC2C(N2CCOCC2C(N)=O)=O)c1 94136,CC(C)C(C)C(CNC(=O)Cc1cnn(C)c1)NC(=O)C=Cc1cncn1C 94137,N1(C(CCc2cccc(C)c2)=O)CCN(C(=O)COC2CC=CC2)C(C(F)F)C1 94138,N1(C(Cc2c(F)ccc(C)c2)=O)CC2CCN(C(C3CC4CC4C3)=O)C(C2)C1 94139,C(CC(=O)NCC(C)CNC(=O)CCNC(C1CCCO1)=O)NC(C)=O 94140,c1(-c2scc(C(=O)NCC(C3CN(C(=O)CNC=O)C3)C)n2)cccc(Cl)c1 94141,c1(C(=O)NC(CCCNC(C(CC)C(C)O)=O)C)ncn2ccccc12 94142,C1(F)(C(=O)NCCCOOCCCNC(=O)Cc2cccnc2)CCOCC1 94143,Cc1cncnc1C(=O)NCCC1(O)CCN(C(c2conc2C2CC2)=O)C1 94144,C1(N(C(C(C2CCOCC2)C)=O)C)CN(C(=O)CCC(=O)N(C)C)CC1(C)C 94145,C1(CC)CN(c2nnc(-c3ccccn3)n2C2CCS(=O)(=O)C2)CCO1 94146,CC(CC(=O)NCCCCCNC(=O)C(F)C1CCCC1)c1ccccc1 94147,C=CCC(C(=O)N1CCC(CNC(=O)CN(S(C)(=O)=O)C)CC1)C(C)C 94148,C1(CCNC(CCOCC)=O)CCCN(C(C2CC(C)(C)C2)=O)CC1 94149,C1(C(=O)NCc2noc(C3CC3)n2)CC(=O)CN1C(=O)CC(O)C1CCCC1 94150,C1(C(C)(C)C)CC(N=c2[nH]c(=NCC=CC3CC3)[nH]c3cccnc23)CCO1 94151,C1(O)(C(N2CC3(C(=O)OCC)C(C2)CCO3)=O)CCc2ccccc2C1 94152,N1(C(c2cc(C(C)C)nc(O)c2)=O)CC2CCC1CN2C(=O)C=CC1CCOC1 94153,C1(C(N2CC(CF)C2)=O)CC2CC1CN(C(=O)CCc1nc(O)n[nH]1)C2 94154,C1(NC(C2CC(=O)NC2)=O)CCOCC1NC(c1cocc1C(N)=O)=O 94155,Cc1ccccc1NC(C1CCCC(NC(=O)Cc2c(C)n[nH]c2C)C1)=O 94156,c1(OCCC)ccc(CNc2ccc(OCCOC)cc2)nn1 94157,Cc1cccc(CNC(=O)C(CNC(C2CC23CCC3)=O)C(C)C)c1C 94158,C1(NC(c2c(OC)cccc2)=O)CN(C(C2CC(C)(C)C2)=O)CC2(CCC2)C1 94159,C(C(CC(C)C)C(=O)N1CCC1CNC(c1cc(Cl)cc(Cl)c1OC)=O)OC 94160,C1(NC(c2cnsn2)=O)CC2CC(NC(c3ccnn3CCF)=O)C2C1 94161,N(C)(C1CCc2c(Cl)cccc21)C(C(N1CCc2c(nc(C)s2)C1)=O)=O 94162,C1(CNC(C2CN(C)C2)=O)CC2CCC1N2C(C1(c2ccccc2)CCOCC1)=O 94163,CCC1CNC(C)C2(CC2)SCC(=O)N1C.C(CC#N)SC 94164,c1(C(=O)NCC2C=CC(NC(=O)CCSC(F)(F)F)C2)sc([N+](=O)[O-])cc1Cl 94165,N1(C(C(CCCCC)C)=O)CCC2(CC1)CC(C(=O)N(C)CC)CO2 94166,CC1CN(C(=O)CCC(N)=O)CC1NC(C1(CC(F)F)CCC1)=O 94167,N1(C(c2n(C)ncc2)=O)CCC(CNC(=O)CC2C=CCC2)CC1 94168,c1(C(=O)NCCN(C(c2ccc(OC)c(Cl)n2)=O)C2CC2)c[nH]nc1S(N)(=O)=O 94169,O=C1NCCn2nc(C(N3CC(CNC(C45CCC(CC4O)C5)=O)C3)=O)cc21 94170,CC1(C)OC2C3CC(C2O1)N(C(c1ccc(OC(F)(F)F)cc1O)=O)C3 94171,N1(C(c2c(OC)cc(C)s2)=O)CCCOC(CCNC(C2CC2[N+](=O)[O-])=O)C1 94172,C1(C(N2CC3CCC2CC3)=O)(N(C(=O)OC(C)(C)C)C2CC2)CC2CCC1C2 94173,C(=O)(C(CC)C(=O)NCCn1cc(C(O)C(C)(C)C)nn1)OCC 94174,C1(NC(C2CC(=C)C2)=O)CCC2CCN(C(c3ccc(-n4cncn4)c(N)c3)=O)C12 94175,c1(C(=O)NC(CC)CNC(=O)CC(=O)OC(C)(C)C)cc(C)c(C)c2ncsc12 94176,N1(C(C(CCC)C#N)=O)CCC(C)(C)CC1C(=O)NC(c1ncc[nH]1)CC 94177,N1(C(C2CCCS2)=O)CCC2OCCN(C(c3nnn4ccccc34)=O)C2C1 94178,C1(COC)CN(C(c2ccsc2)=O)CCN1C(=O)C#CC1(C)CC1 94179,C1(NC(=O)OCC)CCN(C(C2(C)CCCN(C(=O)OC(C)(C)C)C2)=O)C1(C)C 94180,CC1CN(C(C2(F)CCCC2)=O)CC1NC(c1ccnc(CO)c1)=O 94181,C1(O)(C(N(CCNC(c2ccccc2O)=O)C2CC2)=O)CCSCC1 94182,N1(C(CN(C(C(C)C)=O)C)=O)CCOC(CNC(=O)CCC2CCCCN2C)C1 94183,N1(C(=O)CCN2CCC(O)CC2)CC2OCC(NC(C34CC(CO3)C4)=O)C2C1 94184,C1(NC(c2cc(C)on2)=O)CN(C(=O)CC(C2CC2)C2CC2)CC1C(F)F 94185,C(C(=O)NC1CCCCC1NC(=O)CCOC1CCC1)(C(C)C)OCC 94186,C1(C(=O)OC)C(C(=O)OC)C2CCC1N2C(c1ccccc1Br)=O 94187,C(=O)(C(C)CC(F)(F)F)NCCC1(NC(C(C2CC2)OC)=O)CCOCC1 94188,N1(C(C(C)C(C)(C)C)=O)CC(NC(c2nccc(Cl)c2O)=O)CC12CCCCC2 94189,C12(C(=O)NCCCCO)CCC(C(=O)Nc3coc(C4CC4)n3)(CC1)C2 94190,Cc1c(SCC(C(C)C)C(C)C)ccc([N+](=O)[O-])c1[N+](=O)[O-] 94191,C(=O)(CCCCC(C)=O)N1CC(C(N2CCC(F)(CO)CC2)=O)(CC)C1 94192,c1(C(N2C(C)CC(CNC(CC=CC=C)=O)C2)=O)cc(Cl)ncc1F 94193,c1(NC(N2C(C)(C)C(O)C2)=O)cc(C(F)(F)F)ccc1O 94194,c1(OC)c(F)ccc(C(=O)NCC2CCC2NC(c2ccsn2)=O)c1F 94195,c1(C(=O)NC2CCCC(NC(c3c(CCC)n(C)nn3)=O)C2)cc2n(n1)CCO2 94196,C1(C(=O)NC(C=C)C)OCCC1CNC(C1(OC)CCC1)=O 94197,Cc1c(C(=O)NCC(c2ccccc2)NC(C2C(C3CC3)C2(F)F)=O)cccc1O 94198,C1(C#N)(C(N2CC(COC)(NC(=O)CC3CCC4CC34)C2)=O)CCCCC1 94199,C1(C(N2CC(O)C(O)C2)=O)(CC)CCCN(C(=O)CN2CCNC(=O)C2)C1 94200,CNS(=O)(=O)N1CCC(C(N2CCCC2CCNC(=O)CC(C)COC)=O)CC1 94201,c1(N(C)C(=O)NC2CCCN2C(=O)Nc2cnn(C)c2)cc(F)cc(F)c1 94202,Cc1[nH]c(C#N)cc1C(=O)NC1CN(C(=O)C2=CC(C)(C)C2)CC1C(F)F 94203,CCCCC(C(=O)NC1CC(=O)N(C2CN(c3ccc(Br)cc3F)C2)C1)NC(N)=O 94204,c1(OCCC(=O)NCCC(F)Cn2cc(C3CCCCO3)nn2)ccccc1Cl 94205,C1(NC(c2nn(CC)c(O)c2)=O)CN(C(=O)Cc2cnccc2C)CC2(CC2)C1 94206,c1(OC)ccn2cc(C(=O)NC3(C)CN(C(=O)C4=CCCCC4)C3)nc2c1 94207,n1(CC=C)cccc1C(N1CC=CC1CNC(=O)COCc1ccnn1C)=O 94208,C12(C(=O)NC(C)C(=O)NCCF)C(NC(c3cnc(S)nc3)=O)C3CC1C2C3 94209,C1(CC(=O)NCC#CCNC(C2CCN(CC(C)C)C2)=O)COC(C)(C)CO1 94210,C(C)(c1ccccc1F)=CC(=O)NC1CCN(C(c2nccc(CC)c2)=O)C1C 94211,c1(-n2c(CC3COCCN3C)nc(-c3ccc(SC)cn3)n2)ccc(Br)cc1C 94212,C1(C(=O)NCCNC(CN2CC(CC)C2)=O)(C(=O)N(C)C(C)C)CCCC1 94213,C1(CNC(c2n(C)cc(Cl)c2)=O)CCCCN(C(=O)C(C)(C)c2ccsc2)CC1 94214,c1(C(=O)NC(C(=O)OC)CC2CC=CCC2)n[nH]c2c1COC2 94215,N1(C(C(C)(C2CC2)OC)=O)CCC2(CCCCC2NC(=O)C(C)C2CC2)C1 94216,C12(CC(=O)N(C)CCNC(=O)C=CC3COC(C)(C)O3)CCCCC1C2(F)F 94217,c1(C(=O)N(c2ccnc(Br)n2)CCSC2CCCN2)ccc(Cl)cc1 94218,C(c1ccc(Br)o1)=CC(=O)NCC(C)(C)NC(c1ccc(=N)[nH]n1)=O 94219,N1(C(CCCC#N)=O)CCN(C(=O)Cn2ccc3ccc(F)cc23)C2COCC12 94220,C(C)(C)(C(C)NC1(OC)C(C(=O)OC)CC1)NC(C1(C(=O)OC)CC1)=O 94221,C1(CC)CN(C(=O)C(C)C)CCC1NC(=O)C(Cc1cccc(C)c1)N(C)C 94222,CCC(C(=O)NC1CC(CO)N(C(C2CNC(=O)N2C)=O)C1)C(C)C 94223,N#CC1(Nc2cc(Br)ccc2Cl)CCCC2(CCC2)C1 94224,c1(CNc2ccc(NC(C3CC(=O)NCC3)=O)nc2)cn2ccccc2n1 94225,CC(C)CC(CNC(c1cnn(C(C)C)c1)=O)C(=O)NC1CCSCC1 94226,N1(CC)C2CCC1CN(C(C1(NC(C3CCC(C)=C(C)C3)=O)CCOCC1)=O)C2 94227,Cc1cccc(C2(F)CCN(C3CCN(c4cccc(F)c4)C3=O)C2)c1 94228,C1(OC)CC(CNC(c2cncc(C(F)F)c2)=O)N(C(=O)COCC(F)(F)F)C1 94229,Cc1cc(Cl)ccc1OCC(=O)NCCC1=CCN(C(C2CCC(C)O2)=O)CC1 94230,c1(CC)cccc2c1NC(=O)C2NC(=O)OC(C)(C)C.C12(N)CC(C1)O2 94231,C1(C(=O)NC(C)(C)C(N2CCOCC(O)C2)=O)CC(=O)CC12CCC2 94232,c1(C(N2CC(O)(CNC(CC3C(C)(C)C3)=O)C2)=O)nc(F)ccc1Cl 94233,CC1C(C)N(C(C2CCC2)=O)CCN1C(c1cc(C2CCOCC2)[nH]n1)=O 94234,c1(C(c2nnnn2Cc2c(C)n[nH]c2)Nc2ccco2)cn(C)nc1N(C)C 94235,C(=O)(C(CCC1CC1)NC(=O)C(C)SCCCC)NC(C=C)CO 94236,CC(C(=O)N1CCC(CC2CCC2)C1)S(C)(=O)=O 94237,C1(C(N2CCC(NC(C)=O)C2)=O)CCN(C(c2c[nH]c(C(N)=O)c2)=O)CC1O 94238,CC1CN(C(=O)C=Cc2cc(Br)cs2)CC1NC(C1(Cl)CC1)=O 94239,CCCCCCCCCC(=O)N1CCN(C(=O)C(C)C2CCCO2)CC1 94240,N1(c2c(OC)cncn2)CCCC2(C1)CN(c1ncnc3n[nH]c(I)c13)C2 94241,c1(C(N2CCC3(C(C(=O)NCCCCCO)C3)C2)=O)cccc2[nH]ccc12 94242,C1(=O)C(C2CC2)CNC(=O)CN1.C(COCCOC)(C1CC1)COCC 94243,c1(C(N(CCC)CCNC(=O)CC2CC=CC2)=O)coc2c(OC)cccc12 94244,c1(C(=O)OC)ccc(C)cc1SC.n12cc(nn1)NCCN(C)CC1CC1C2 94245,Cc1ncc(N)cc1C(=O)NCCOCCNC(C12CCCCC1C2)=O 94246,c1(C(N2CCCC2C)C(=O)NCCCSC)cc(C(F)(F)F)ccc1C 94247,N1(C(c2c(C)c(C(N)=O)ccc2)=O)CC2CC(NC(c3n[nH]cc3Cl)=O)C(C2)C1 94248,c1(C(CNC(C(c2ccccc2)OC)=O)NC(=O)C=CC2CCC2)cnn(C)c1 94249,c1(C(c2nc(-c3cccnc3C)no2)OC)ccc(C)c(F)c1 94250,c1(CC(=O)NCC2C(OC)C3(C2)CCC3)ccc([N+](=O)[O-])c(N)c1 94251,Cc1cnccc1CN(C(=O)CC1CCN(C(=O)C(N2C(C)CC2(C)C)=O)C1)C 94252,C1(C(N2CCC(CC(C)NC(=O)C3CC3)CC2)=O)CCCCC1(C)C 94253,Fc1ccc(N2CCN(CCCC3CC3)CC2)cc1 94254,Oc1ncccc1CN(Cc1ccccc1)CC1CC1C1CC1 94255,Cc1cc(C(=O)NC(C)CNC(C2(c3c(C)cccc3C)CC2)=O)c(N)c(Cl)c1 94256,Cc1cccc(CC(=O)NCCC2(NC(C3CCCC3C(F)F)=O)CCC2)c1 94257,c1(NC(C)=O)cccc(C(N2CC(C(C)NC(=O)C(C)c3ccsn3)C2)=O)n1 94258,Cc1cc(N2CCC(C(N3CC(CNC(=O)C(C)C(C)O)C3)=O)C2=O)ccc1F 94259,c12ncc(cc1Cl)n2C.C1(NC(C)C)CNC(=O)C1.C12(CC1)CCCNC(=O)N2C 94260,C(=O)(CC(O)CN(C)C)N(CC)CC1CCS(=O)(=O)C1 94261,N1(C(CC2(OCC)CCC2)=O)CCCCC1CCNC(C1CC(N=[N+]=[N-])C1)=O 94262,Cc1oc(C(=O)NC2C3CN(C(c4cnc(O)n4C)=O)CC23)cc1S(C)(=O)=O 94263,N1(C(C(CC=CC)NC(c2ccn(C)c2)=O)=O)Cc2nc(C)sc2C1 94264,n1(CC(=O)NC(CNC(C2(OC)CCCOC2)=O)(C)C(C)C)ncc(O)nc1=O 94265,c1(C(N(C2CN(C(C3CC(CF)C3)=O)C2)C)=O)sc(Cl)cc1Br 94266,S(=O)(=O)(c1ccc(NCc2csc(N(C)C)n2)c(Cl)c1)NC(C(CC)CC)=O 94267,C=C1CCN(C(=O)CCOCCCOCC)C(C(=O)Nc2ccc(F)cn2)C1 94268,c1(C(N2CCC(OCCNC(C3CCC3)=O)C2)=O)cnc(C2CC2)nc1 94269,C1(NC(c2cc(C)[nH]c2C)=O)CC(O)CN(C(C2CCC(C)O2)=O)C1 94270,n1(C(CC)CC)nc(C(=O)N(C(CCC(=O)OC)C(=O)OC)C)ccc1=O 94271,N1(C(CC2CCN(C(c3ccc(NC=O)cc3)=O)C2)=O)CCCN(CCO)CC1 94272,C1(C2CN(C(c3ccsc3)=O)C2)(NC(c2cnc(-n3cccn3)cn2)=O)CC1 94273,c1(C(C)(C)C)ccc(C(=O)NCC(C)(CO)NC(C23CCC2C3)=O)nc1 94274,N1(C(COc2ccc(C#C)cc2)=O)CC(C)CN(C(C2(C)CC=CC2)=O)CC1C 94275,C1(OC)CC(CNC(c2cc(F)cs2)=O)N(C(=O)C(n2cc(Cl)cn2)C)C1 94276,C(=O)(CCS(=O)(=O)C(F)(F)F)NC(C(C)(C)C)CNC(C1CCCCN1N=O)=O 94277,C1(C(=O)NCCCN(CC)CC)(CC)CCCN1C(c1n[nH]cc1C)=O 94278,CC1(C(=O)NCC2(NC(C3CCS3(=O)=O)=O)CCCC2)CCC(O)CC1 94279,C1(NC(C(COCC)C)=O)CN(C(c2cc(C)c(Br)o2)=O)CC1SC 94280,CC1(C)CC(C(=O)NCC2CN(C(=O)CCC3CCC3)C(C)(C)C2)CNC1=O 94281,N1(C(C(C)SCC)=O)CC(NC(C2Cc3nnc(C)n3C2)=O)CC12CCOCC2 94282,C1(CNC(c2c(C)ncnc2)=O)CN(c2nc3ccccc3s2)CC2(CCC2)O1 94283,C1(OC)CC(CNC(c2nncn2CC#N)=O)N(C(=O)C(C)OC2CCCC2)C1 94284,N1(C(Cc2c(OC)cccc2Cl)=O)CCCC2(CCc3ccccc32)C1 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94303,C1(CC#C)(C(N2CCC2(C)C)=O)CCN(C(C2CC2Cl)=O)C1 94304,c1(CN(C2CCOC2C)C(C)C)ccc(C(F)F)cc1 94305,C(=O)(C(C)(CC)CC)NC(C(=O)NCCCCOCC)CCC1CCC1 94306,C1(CC(=O)N(CCN=[N+]=[N-])C)C=CC(NC(=O)CCn2cccn2)C1 94307,C1(CC(=O)NCC(C)(C)OC(F)F)CC(C)(C)CN1C(C1CC(=C2CCC2)C1)=O 94308,N1(C(C2N(C(c3c[nH]nc3Cl)=O)CC23CCCC3)=O)CCCC(C2CC2)CC1 94309,c1(C(N2C(C)(CNC(C3=C(C)CCC3)=O)CCC2)=O)cc(Cl)c2ccccc2n1 94310,C(CS(=O)(=O)CC(=O)N1CCCC(n2cc(CNC(C3(C)CC3)=O)nn2)C1)OC 94311,n1(CCC)ncc(C(N2CCCC(CNC(=O)CC=CC3CC3)C2)=O)c1C(F)F 94312,c1(C(=O)NCCCN(C(C2(COC)CCCO2)=O)CC)ccc2n[nH]cc2c1 94313,C1(NC(CCC)=O)CCN(c2cc(-c3ccccc3)ncn2)CC1OCC 94314,c1(C(=O)NCC2C(NC(CCCCC(C)C)=O)C2)cc(F)cc2cnccc12 94315,CCC(CC(C)C)C(=O)NC1CCC1NC(C1(N(C)C)CCCC1)=O 94316,N1(C(C2C(OC)C2)=O)CCN(C(=O)Cc2csc(Br)n2)CC(O)C1 94317,N1(C(c2cnc(C(C)O)s2)=O)Cc2c[nH]nc2C(C)(C)C1 94318,Cc1cc(C(=O)NC2CCCC(C(=O)NOCC3CCCCC3)C2)nc(C)c1 94319,CCC(C)(CCC(C)C)C(=O)N1CC2OCCN(C(=O)C=CC(C)(C)C)C2C1 94320,c1(CNC(C2CCN(C(C3C(C(=O)OC)C3)=O)CC2)=O)cc(=O)n2ncsc2n1 94321,c1(OC)cc(N(C)C)ccc1C(=O)NCC1CC(NC(C2(CO)CC2(F)F)=O)C1 94322,C1(CCNC(c2c(CC)non2)=O)CCCN(C(c2cnc(OC)nc2)=O)C1 94323,N1(C(CCN(CC)CC)=O)CCC2(NC(=O)CCOCC(C)(C)C)CCCCC12 94324,C1(C(=O)OC)(OC(C)=O)CCN(C(=O)C(C)(C)Br)CC1.N12CC(C1)C2=O 94325,c1(-n2c(Cc3nc(C)sc3C)nc(C(C3CC3)OC)n2)cc(CO)ccc1C 94326,CC(C)(CCCC(=O)N1CC2(CCCCC2)C1)NC(=O)Cn1cccn1 94327,C1(CNC(c2nc(-c3ccc(Br)cc3)ns2)=O)CCCN(c2ncccn2)C1 94328,c1(C(N(C)CC2N(C(C(C)C3CC3)=O)CCOC2)=O)cnn2c1CCC2 94329,CCC(C#N)(CC)C(=O)NCC(N1CCN(C(c2cc(C)ncc2C)=O)CC1)C 94330,c1(CCCC(=O)NCCNC(C2COCCO2)=O)c[nH]c2ccccc12 94331,C1(C(=O)NCc2cc(OC)ns2)CN(C(=O)C=CC2CCCC2)CCN1C 94332,N1(CC)CC(C(N2CCC(CC(C)NC(=O)C(C)(F)F)CC2)=O)CCC1=O 94333,c1(C(N2CCC(O)(CN(C(=O)CN3CC4CC4C3)C)C2)=O)ccc(F)c(O)c1F 94334,c1(CC(=O)N(C)CC2CCN(C(C(COCC)C)=O)C2)ccc(F)cc1 94335,c1(NC(C(=O)NC2(CN(C(CC(C)C)=O)C)CC2)=O)ccc(C#N)c(Cl)c1 94336,N1(C(c2cc(C)oc2)=O)CCC(NC(c2cnn(C)c2)C)C(C)C1 94337,c1(OCCCC(=O)NC(CNC(CC=CC)=O)COC)ccc2c(c1)CCC2 94338,n1(CC)cccc1C(=O)NCCC1(NC(=O)C=CC2CCCO2)CCCC1 94339,C1(N(C(c2c(C)occ2)=O)C)CCCC2CN(C(c3ccc(=O)n(C)c3)=O)CC12 94340,C1(NC(CSCC#C)=O)CC2CN(C(=O)C(C)CC3CCCC3)CC2C1 94341,C1(C(=O)OC)CCN(C(=O)CSc2cc(Cl)ncc2OC)CCC1(F)F 94342,c1(CC(=O)NC2CN(C(c3csc(C4CCCC4)n3)=O)C3CC23)cccnc1O 94343,C12(C(=O)NCCNC(C3(C(=O)NC)CC3)=O)CC(c3ccccc3)C1C2.CO 94344,O=C1C=C2CN(C(C34CC(C3)C4)=O)CCC2S1.C12COCCN1C2=O 94345,c1(C(N(C(C)CNC(c2cccc(Cl)c2OC)=O)CC)=O)cc(Cl)cc(C)c1N 94346,c1(C(=O)NCC(=O)NC(C(=O)OC)Cc2cn(C)cn2)cccc(Br)c1 94347,N1(C(c2cc(C3(C)CC3)on2)=O)CC2CN(C(C3CCCN3N=O)=O)CCC12 94348,Cc1ncsc1CCC(=O)NC1CC(CCNC(C2(CO)CCC2)=O)C1 94349,C(CCC(O)C(=O)NCCOc1ccccc1)NC(Cn1nc(C)oc1=O)=O 94350,CC(C)S(=O)(=O)CC(=O)NC1CC(CCNC(c2ccc(N(C)C)cc2Cl)=O)C1 94351,C1(C(=O)NCc2c(OC)nccc2)CC2(CC(NC(=O)C(C)S)C2)C1 94352,C(C)(C(=O)NNC(=O)N1CCCC1CO)n1cc(Nc2ccc(OC)cc2)nn1 94353,O=C(CCC(F)(F)F)NCC1(CO)CCN(C(C2CCCC3(CC3)C2)=O)C1 94354,N1(C(c2cc(C)on2)=O)CCN(C(C2COC3COCC3O2)=O)CC(O)C1 94355,N1(C(c2ccc(C(C)=O)cc2)=O)C2CCC1CC(NC(c1cc(Cl)cnn1)=O)C2 94356,C1(NC(C2CC(OC)C2)=O)CCCC2CN(C(=O)CCn3c(C)csc3=O)CC12 94357,c1(C(=O)NCC2(O)CN(C(=O)CC3CCC(O)C3)C2)cnc2c(c1)COCC2 94358,C(=O)(CCCCCN(C(=O)C(C)SCC)C)N1C(C#C)CC1 94359,C1(NC(c2cc(CC)ncc2)=O)CC2(CCCCN2C(C2CC=C(C)CC2)=O)C1 94360,C1(C(=O)NCc2cscn2)CC2(C1)CN(C(=O)C(c1ccccc1)O)C2 94361,Cn1ncc2c(NCc3cc(Cl)cc(Cl)c3)[nH]c(=NCCCC(F)(F)F)nc12 94362,C12(CNC(C(CC)SC)=O)CCCC1CN(C(c1ccn3ccccc13)=O)C2 94363,c1(C(=O)NC2C(NC(C3C(CCC)C3)=O)CCC2)cn(C)[nH]c1=N 94364,N1(C(C2CCC(SCC)CC2)=O)CC2CCC(NC(C3CC4C=CC3C4)=O)C2C1 94365,c1(C(=O)NCC(C)CNC(C2CC3CCCC(C2)C3)=O)cc(N)c(N)cc1F 94366,C1(C(=O)NCC2(CCNC(c3cc(-c4ccoc4)[nH]n3)=O)CC2)CCCCS1 94367,c1(CNc2cc(C(F)(F)F)c(Cl)cc2)cccc2sccc12 94368,c1(C(=O)NC(CCCC)CNC(C2C(C)C2C)=O)cccn2ncnc12 94369,CCCCCCCC(=O)N1CCC1CNC(c1ccc(C(C)(C)C)nc1)=O 94370,c1(C2(C(F)(F)F)CCSCC2)nnc(C2CCc3cccc(Cl)c32)o1 94371,c1(CNC(CCCCN(C(c2c(COC)n[nH]c2)=O)C)=O)cc(C)cnc1F 94372,C(CC(O)C(F)(F)F)NC(C=CCN(C(CCCOCC=C)=O)C)=O 94373,C1(C)(CNC(C(C)SC)=O)CCN(C(c2cncc(CO)c2)=O)C1.C(N)=O 94374,CC(=O)C(C)CC(C)C(=O)N1CCC(C)(C)C1C(=O)NOCC(O)CO 94375,C1(C2(OCC)CCC2)(NC(CC2CCCN(C(C(CCC)=CCC)=O)C2)=O)CC1 94376,N1(C(C)C(=O)NCC(c2ccccc2)NC(=O)CC2CCC2)CCC(O)CC1 94377,c1(NC(=O)NC2CCN(C(=O)C=Cc3ccccc3)C2)ccc2cccnc2n1 94378,N1(C(=O)OC(C)(C)C)CCCC1CNC(C1CC(N2CCCC2)C1)=O 94379,Cn1cnc2sc(C(N3CC4CC3CN4C(=O)CC3CCC(F)(F)C3)=O)cc12 94380,c1(COc2ccc(C(CC)C)cc2)cnc2[nH]ccc2c1 94381,N1(C(COC)=O)CC(NC(c2sc3cccc(F)c3c2C)=O)CC12CCOCC2 94382,c1(OC)ccc(C(F)F)cc1NC(=O)C(=O)NCCC1CC(=O)C12CCC2 94383,c1(OC)cc(NC2CCC(NC(=O)C(C)CN(C)C)CC2)ncn1 94384,C1(C(N(CCF)CC)=O)CC(NC(C2CC(F)(CF)C2)=O)CCO1 94385,n1(C(CC)C)ncc(C(=O)NCC23CC(NC(c4ncnn4CC)=O)(C2)C3)c1C 94386,C(C(O)CC(C)(C)C)NC(C1CC(O)(CNC(c2n(CC#C)cnn2)=O)C1)=O 94387,c1(C(=O)NCC(C2CCC2)NC(c2c(C)snc2)=O)cnn(C)c1Cl 94388,C(=O)(CC(C)C(C)C(C)C)NC(CC)(CC)CCNC(c1cn(C)ccc1=O)=O 94389,C=CCCC(O)CNC(C12CC(CN1C(C1(C(C)(C)OC)CC1)=O)C2)=O 94390,C(CCCCC(=O)NC1(CF)CCN(C(=O)CC(=O)OCCC(C)C)C1)SC 94391,c1(OC(CC)C#N)cc(NC(=O)C(N2CCC(CN(C)C)CC2)=O)ccc1OC 94392,Cc1ccc(S(=O)(=O)N2CCC(O)(C(=O)Nc3ccc(Br)nc3)CC2)c(C)c1 94393,CC1CCN(c2ccc(NC(=O)NC3(CC4CCC4)CC3)cc2)CC1 94394,Cc1cncc(OCC(=O)NC(C2CCCN2C(=O)C2=CCSC2)(C)C)n1 94395,N1(C(C2CN(C(CCOCC#C)=O)CC2C(C)C)=O)CCCC(C)(F)C1 94396,C(C(COC)C(=O)N(CC(C)(C)CNC(=O)CC1C=CCCC1)C)OC 94397,CC(C)C#CC(=O)NC1CCC(N(C(=O)CC2CCCO2)C)CC1 94398,C(=O)(C(F)(F)C(C)O)N1CC(C)(CCC(=O)NCCN(C)CC)C1 94399,N1(C(C)CNC(c2cnccn2)=O)CCN(C(=O)CN2CCC(C)(C)C2)CC1 94400,C1(CCC)(CNC(=O)CCCN(C)C)CCN(C(C2(CCOC)CCC2)=O)CC1 94401,C=CCCCC(=O)N1CCC(N(C(=O)C(C)Cc2cnn(C)c2)C)C1 94402,N1(C(C23N(C(C(C)OCC(C)C)=O)CCC2C3)=O)CC(C)(C)OC(C)(C)C1 94403,C(=O)(CCC1=NNC(=O)CC1)N1CC2(OCC(NC(C(CCC#C)O)=O)C2)C1 94404,c1(OC)cccc(C(=O)NC(C)CCN(C(=O)C(C)(C)C2CCCC2)C)n1 94405,CCCC(CC)C(=O)NCC1CCCN(C(c2cncc(CO)c2)=O)CC1 94406,C#Cc1ccc(C(=O)NCC2CCCN2C(=O)C(C)CN2CCOCC2)cc1F 94407,CC1CNC(=O)CC(NCc2ccc(Cl)c(Cl)c2)C1 94408,c1(C(=O)NC(CNC(CN2CCCC(CC)C2)=O)CO)cccc2c1CCN2 94409,C1(NC(C(CO)OC)=O)CCCC(C(=O)NCC2(c3ccon3)CC2)C1 94410,Cc1cc(C(=O)NC2CC3(C2)CN(C(c2cc(C)sn2)=O)C3)c(O)c(C)n1 94411,C1(NC(C2(C)C=CCC2)=O)C=CCN(C(=O)Cc2ccnc(Br)c2)C1 94412,Cc1ccc(CN(CC(N2CC(NC(C3CCCC3(C)C)=O)C(C)C2)=O)C)cc1 94413,C1(OC)CCC2(C(N3CC(NC(=O)C(C)OC4CCCC4)C(C)C3)=O)CC12 94414,C12(NC(c3cncc(OC)c3)=O)CCCN(C(c3ccsc3C(F)F)=O)CC1C2 94415,c1(C(=O)NCCN(CC(C)O)C(=O)CC2CC=CCC2)ccc(Cl)c(N)c1 94416,N1(C(c2ccc(SC)cc2)=O)CC2CC1CCN2C(=O)C=Cc1nc(C)cs1 94417,C#Cc1cncc(C(=O)NC(C)C(c2c(F)cccc2F)O)c1 94418,C(c1ccc(F)cc1)=CC(N1CC2CN(C(C3CCCS3)=O)C2C1)=O 94419,N1(C(c2cn(CC)nc2C2CC2)=O)CC2(CC(NC(C3CCNC3=O)=O)CO2)C1 94420,C(=O)(C1=C(C#N)CCC1)N1CCC(C=C)(C(=O)NCC(C)N(C)C)C1 94421,C(=O)(C(C)(C)CC(F)(F)F)NCC1N(C(CCCc2n(C)cnn2)=O)CC=C1 94422,c1(CN(C2(C(=O)NC(C)=O)CC2)C(=O)Cc2cnoc2)ncnc2ccsc12 94423,Cc1cc(F)cc(C(=O)NC2CCC(NC(=O)C(O)C3CCCC3)CC2)c1C 94424,Cc1cc(F)c(NC(=O)NCCC2CCCN(C)C2)cc1Cl 94425,CC(C)(O)CCNC(=O)CC1(NC2CCN(Cc3ccccc3)C2)CCC1 94426,N1(C(c2nc(C)sc2)=O)CCCC(C)(C(=O)Nc2c(Cl)c(C)nn2C(C)C)C1 94427,N1(C(C=C(C)C(C)(C)C)=O)CC2CC1C2C(=O)N(C1CCCC(O)C1)C 94428,C1(C)(CNC(C=NOC)=O)CN(C(=O)COC2CC=CC2)C(C)(C)C1 94429,C1(C(=O)NC2CCC(CNC(CC(C)(C)OC)=O)C2)Cc2ccccc2C1 94430,N12CC(CCC1C)NC(=O)C1C(CCC1)C2=O.C1(C(=O)OC)(OC)CS(=O)(=O)C1 94431,C1(C)(C(=O)NC(C2N(C(c3c(C)snn3)=O)CCC2)C)CCN(C)C1=O 94432,C#Cc1ccc(NC(=O)CC2(c3ccc(OC)cc3)CCC2)cn1 94433,C(C(C)(C)C(=O)NC(c1ccccc1F)CNC(C1CCCO1)=O)N(C)C 94434,S(=O)(=O)(c1ccccc1C(F)(F)F)N1CCC(F)(CNS(CCCC)(=O)=O)CC1 94435,C1(NC(c2c(C)cc(F)s2)=O)CC2CCC(C1C)N2C(c1ccc(CO)cc1)=O 94436,C1(CC(=O)N(CCCNC(=O)C(O)Cc2cnc[nH]2)CCC)CCCCC(=O)N1 94437,C1(NC(CCC(C)=O)=O)CCN(C(c2ccc(C(F)(F)F)nn2)=O)C(C)C1 94438,c1(SC)cc(F)ccc1C(=O)NC(C)CCCCNC(C12CCC(C)(CO1)C2)=O 94439,C12(CNC(C(COC)(F)F)=O)CCCC1N(C(c1c[nH]c(=N)s1)=O)CC2 94440,C#CCC(CC(F)F)C(=O)NCc1ccc(CNC(=O)CCC(=O)NCC)cc1 94441,c1(C(=O)NCC(CC(C)C)NC(=O)C(C#N)=CC2CC2)cccc([N+](=O)[O-])c1 94442,C1(N(C(CC)=O)C)CCCC(NC(=O)Cn2nnnc2C)C1 94443,c1(CC(=O)NC(C)(C)CN(C)Cc2ccnc(SC)n2)c[nH]c2ccccc12 94444,CC1CCCN(Cc2ccccc2F)C1NC1CCN(C(c2ccccc2)=O)CC1 94445,c1(NC2CC(C)N(C(=O)Cc3ccc(Cl)s3)C2)nc2c(cc1C#N)CCC2 94446,c1(C(=O)NC(C2CCOC2)CNC(c2cnc(OC)s2)=O)cccc2c1CCO2 94447,c1(C(=O)Nc2ccc(OC)cc2)c(C)o[nH]c1=NC(=O)c1nnn2c1C(=O)NCC2 94448,c1(C(=O)NCC2C(C)CN(C(=O)Cc3cccc(Cl)c3)C2)ccnc2[nH]cnc12 94449,N1(C(CCCC)=O)CC(CNC(=O)CNC(c2ccc(C)s2)=O)C(C)C1 94450,C1(C(N)=O)(OCc2ccccc2)CC(O)C12CCC2.N12CCC(CC1)CNC2=O 94451,N1(C(c2c(C)cc(C)[nH]2)=O)CCCN(C(=O)COCc2ccccc2)C(CO)C1 94452,C12CCN(CC1)CCN2C(=O)NC.c1(NC(C2(CC=C)CCC2)=O)ccc(Br)o1 94453,c1(NC(N2CCC(C3CCC(N(C)C)O3)CC2)=O)cccc2c1CCCC2=O 94454,c1(C(C)NC(C2(F)CN(C(C(C)SC)=O)C2)=O)cncc(F)c1 94455,C(=O)(C1=COCCC1)NCCC(C)O.C12CCC1C(=O)N2 94456,C1(CCC)CC(C(=O)NCC2CCCCN2C(=O)Cc2cccs2)CCO1 94457,c1(N(CCCc2ccccc2)C)nc(=N)[nH]c(=NC2CC2C2CCC2)[nH]1 94458,CC1(C)CCOC1C(N1CCC(C)(CC(=O)NC(c2ccncc2)(C)C)C1)=O 94459,C(=O)(C(C(=O)N1CC2(CNC(=O)Cn3ccc(C)n3)CCC1C2)C(C)C)OCC 94460,c1(C(N2C(CNC(C(C)(O)C3CC3)=O)CCCC2)=O)cnc(Cl)cc1Cl 94461,C1(NC(c2nc(C(C)OC)oc2)=O)CCC(NC(C2CC2F)=O)CC1 94462,c1(C(=O)NC2CC2NC(C2CC(=O)N(C3CCCC3)C2)=O)csc2c1CCCC2 94463,CC1CN2CCN1CC2C(N1CCC(C)(CNC(=O)C(c2ccccc2)=O)C1)=O 94464,N1(C(CC(CC)CN(C)C)=O)CCC(N=c2nc(C(F)(F)F)[nH]s2)C2(CCC2)C1 94465,CC#CCC(C(=O)NCCC(C)CC)NC(=O)C(=O)N(C)C 94466,N1(C(CNS(CC)(=O)=O)=O)CCCC(CCNC(C2CCCO2)=O)CC1 94467,c1(OC)ccc2cc(C(N3CCC4CN(S(=O)(=O)CC(C)C)CC34)=O)ccc2c1 94468,c1(OC)nc(C)ccc1C(N1CC(NC(=O)Cc2nnc(C)o2)C(C#N)C1)=O 94469,Cn1cnc2c[nH]c(=NCCC3CCN(C(c4ccc(C(N)=O)nc4)=O)C3)nc12 94470,N12CC3CN(CC3C1)CC2=O.C1(CCC(=O)NC2CC3(CC3)C2)CCCCC1 94471,C(=O)(CCCCCCCC1CC1)NCC(C)NC(c1c(C)ccs1)=O 94472,N1(C(C2C(=C)C2)=O)CCCC2(C1)C(NC(=O)C(C(F)(F)F)C(F)(F)F)CCN2C 94473,C1(CC)CCCN(C(=O)CC(C)(C)C2CC2)C1C(=O)NC1CN(C)C(C)(C)C1 94474,CC1CCCC=C1C(=O)N1CC2(CCCC2NC(c2cnc3nccn3c2)=O)C1 94475,CC(C)S(=O)(=O)c1c(C(=O)NCC2CC3(CCN2)CCOCC3)cccc1Cl 94476,CCC1=C(C(=O)NCC2CN(C(=O)C(C)c3ccco3)CCO2)CCCO1 94477,Cc1cc(SCC(=O)NCC(C)(CO)NC(C2CC(C)CCO2)=O)cc(C)c1 94478,c1(C(=O)OC)cc(OC)cc(OC)c1CC(c1ccccc1)=CC1CC1 94479,CCC(CC(=O)NC1CC1CNC(=O)CN(C)C(N)=O)C(C)C 94480,c1(C(N2C(CNC(c3c(C)[nH]c(C(F)(F)F)c3)=O)CC2)=O)cc(S(N)(=O)=O)co1 94481,C(=O)(C(C)CCCOC)NC(CCCCNC(CN(CCCCCC)C)=O)C 94482,c1(C(=O)NC(CC)(C)CNC(c2ccc(C(F)F)o2)=O)c(C)cc(C#N)cc1C 94483,n1(CC)nc(C)c(C(=O)NCC(C)N(C)C(c2sccc2C#N)=O)c1C(F)F 94484,N1(C(C(=O)N(C)C)=O)CCN(C(=O)C(C2CC2)NCc2ccc(CO)cn2)CC1 94485,c1(NC(=O)C(=O)NCc2cscc2Br)ccc(CCOCC(=O)N(C)C)cc1 94486,C1(C(=O)NCC2CN(C(Cn3nc(C)oc3=O)=O)C2)Cc2ccccc2C(=O)O1 94487,[N-]=[N+]=NC1CC(C(=O)NC(CO)CCF)N(C(=O)C#CC2CCC2)C1 94488,N1(C(C(C)N(CCC)C(c2csc(Cl)c2)=O)=O)CC(=O)N(C)CC1C 94489,CC1CN(C(C2CN(C(=O)CCC3(C#N)CCC3)CCO2)=O)Cc2c[nH]nc21 94490,c1(C(N(C(C(C)C)Cc2ccc(F)cc2)C)=O)ccc(N2CCCC2=O)c(Cl)c1 94491,Cc1ccc(-n2nc(CCSc3ccccc3)nc2-c2ccccc2F)c(C)c1 94492,CC1(C(=O)NCC2OCCC2C(=O)NCCOCC2CCC2)CC(C#N)C1 94493,Cc1cccc(Br)c1C(C(=O)N(CC(C)C(C)(C)C)C)NC(c1c[nH][nH]c1=N)=O 94494,C=CC(CC)CC(=O)NC12CC(C1)N(C(=O)C(C1CC1)OC)C2 94495,C=CCCCCCC(C)(c1nnnn1CCCOC)NC(C)CCCC(C)C 94496,C(C)(C)(CN=c1[nH]c2ccccc2s1)C1CCN(C(C(C)OC2COC2)=O)CC1 94497,C1(C(=O)NC(C)CNC(=O)CCc2cncc(F)c2)Cc2nn(C)cc2C(=O)N1 94498,C12(C(N3C4(CNC(c5c(C)scn5)=O)CC(C3)C4)=O)CC(C)(C1)OC21CCC1 94499,CCC1=NOC(C(=O)NC(CNC(c2cnn(CC)c2C2CC2)=O)CC)C1 94500,C1(C(=O)NC2CC(NC(c3c[nH]c(=NC)s3)=O)C2)CCc2c[nH]nc2C1 94501,Cc1cc(C(F)F)oc1C(N1CC(N(C)C(C2CCC(F)(F)C2)=O)C(O)C1)=O 94502,CN1CCOC(C(=O)N(C)CC2COCCN2C(c2csc(Cl)c2)=O)C1=O 94503,C1(CC(N2C(C(CNC(COC(CC)(C)C)=O)O)CCC2)=O)COCCN1CC 94504,Cc1csc(C(N2CCCC(C(C)NC(C34CC(CCO3)C4)=O)C2)=O)c1C 94505,C1(C(=O)NC(c2cn(C)nn2)C(=O)NC(CC)CCCO)CCOC(=O)CC1 94506,c1(OC)ccc(C(C)(C)C(=O)N(CC(O)CN(C)C)C)cc1OC 94507,C1(CNC(=O)C=Cc2cnc[nH]2)CC2(CC2)CN1C(=O)CC1COC2CC1C2 94508,C1(CCC)CN(C(=O)CC(C)CC)CCN1C(=O)CN1CCC(C)CC1 94509,C1(CCC)(NC(=O)CCC2CC2C)CCN(C(C2CC3CCC3C2)=O)CC1 94510,c1(C(=O)NC2C(CNC(c3cc(CC)ns3)=O)CCC2)cc(CC)nn1C(C)C 94511,N1(C(C2CC(CF)C2)=O)CCC(Cn2cc(C3COCC3O)nn2)C(F)(F)C1 94512,CCCC(CC)C(=O)NC1(CO)CCCN(C(c2cc(C(CC)CC)no2)=O)C1 94513,N1(C(c2cc(C)c(N)cc2F)=O)CCCC2(CC(NC(c3ccoc3)=O)C2)C1 94514,C(=O)(CCC(F)(F)F)N(CC(C)NC(=O)C(C)CC1CC1)CC 94515,C1(C(=O)NC(C(N2CC(C#C)C2)=O)Cc2cn[nH]c2)CC12CCCC2 94516,C(=O)(CCCC(=O)OC(C)C)N(CCCNC(C(COC)OC)=O)C 94517,c1(CN)ccccc1-c1cn(CCC(=O)NC2CC3CC3C2)nn1 94518,C1(CC(=O)NCC(C)C2CC2)CC(NC(C2CCCC2)=O)C1 94519,n1(CC(=O)OC(C)(C)C)cccc(Nc2cccc(CC(=O)O)c2)c1=O 94520,c1(C(N2CC3CC2CCC3NC(=O)C(F)(F)CC2CC2)=O)cccn2ccnc12 94521,N1(C(C(C)(C)NC(=O)OC)=O)CCC(C2CC2)(CNC(=O)C=CC(N)=O)C1 94522,C1(C)(CNC(C(C)OCCC=C)=O)CCCN(C(c2cn(C(F)F)cn2)=O)C1 94523,O=C(C1CCCOc2ccccc21)NC1COCC1n1cc(-c2ccsc2)nn1 94524,c1(CNC(c2c(C)cnn2C)=O)ccc2c(c1)CCC2NC(=O)CSC(F)(F)F 94525,c1(C(=O)NC(C2(CNC(C3CC(SC)C3)=O)CC2)C)cc2ccncc2c(O)n1 94526,N1(C(CCSCCCC)=O)CC2CC2(NC(c2oncc2C)=O)C1 94527,C1(OCc2cccnc2)CCN(C(=O)CN(C(C2C3CCC23)=O)CC)CC1.C1CS1 94528,N1(C(c2nn(C)c(F)c2)=O)CCCCCC1CNC(C1C2CCCCC12)=O 94529,c1(C(N2C3(CNC(C(CC)F)=O)CC(C2)C3)=O)nc(C(C)C)ncc1Br 94530,C1(C(F)(F)F)CCC(F)(c2nc(C34CC5CC3C4C5)no2)C1 94531,c1(C(=O)NC2(c3ccccc3)CN(C(C3C4COCC34)=O)C2)n[nH]c(O)n1 94532,c1(C(=O)NC2CC3(C(NC(CC4ON=C(C)C4)=O)C3)C2)ccnc2[nH]c(O)nc12 94533,n1(CC(N2CCCCCC(NC(C(C=C=C)C)=O)C2)=O)[nH]cc2c(=O)ncnc1-2 94534,C1(C(=O)NCC(CNC(CC(C)OC)=O)O)CC(=O)N(C(C)C2CC2)C1 94535,CCCCC(CC)C(=O)NCC(C)(C)NC(c1sccc1SC)=O 94536,Cc1cc(C(N2CCNC(C(=O)NC3CC(O)C3)C2)=O)cc(C#N)c1 94537,c1(C(=O)NCCC2(O)CN(C(CSCC)=O)C2)sc2cncn2c1C 94538,c1(CNC(C2CCN(CC(C)(C)C(=O)O)CC2)=O)ccc(F)c2[nH]ncc12 94539,N1(C(C(CCNC(C2(CC3CCC3)CC2)=O)OC)=O)CCCC(C)(O)C1 94540,C1(NC(CC)=O)CCCC12CCN(C(=O)COc1ccc(F)c(F)c1)CC2 94541,c1(C(N2CCC(F)(CO)CC2)=O)cccc(F)c1-c1cnc(F)c(OC(C)C)c1 94542,c1(C(=O)NC(c2cccc(N)n2)C)cnc2n1CCOCC2 94543,C(=O)(C(C)(C)CC(F)(F)F)N(CC(CNC(c1c(OC)n(C)nc1)=O)C)C 94544,CCC(C)(O)C(=O)NC1C=CCN(C(c2cn(C)nc2C)=O)C1 94545,c1(CCC(=O)NCC(CCNC(CCCOC)=O)OC)ccc(O)cc1 94546,CCC(CC)C(F)C(=O)NC(CC1CCCC1)C(=O)N(C1CCC(F)(F)C1)C 94547,C1(CC(=O)NC(CN(C(=O)CCCCSC)CC)C)COCCN1C 94548,C12(C(=O)NC3CC(F)(CNC(c4c(C)ncs4)=O)C3)CC(C)(CO1)C2 94549,C(CN=c1[nH]c2c(c(=NC3CC4(C3)CC43CCC3)[nH]1)COCC2)OC(C)(C)C 94550,Cc1cc2ncc(C(=O)NCC(C)NC(=O)CN3CCCC3C)cc2[nH]1 94551,N1(C(CCC=C)=O)CCC(CO)(NC(=O)Cc2csc(-c3cnccn3)n2)C1 94552,c1(C(N2C(CC(=O)OC)CS(=O)CC2)=O)cc(Br)c(C(F)(F)F)cc1F 94553,C1(CNC(=O)C(O)CN2CCOCC2)CCN(C(c2cc(CCO)on2)=O)CC1 94554,N1(C(CCN(C(C)=O)C)=O)CCC(CO)(CNC(=O)CCCC2CCOCC2)C1 94555,c1(CNc2ccc(OC)c(Br)c2F)cnc2c(c1)c(C)nn2C 94556,C(=O)(C(C1CN(C(C2(CN(C)C)CC2)=O)C1)OC)N(CC(=O)OCC)CCC 94557,C1(NC(C(=O)NC(CC)CC(C)CO)=O)CC2COCC2N1Cc1ccccc1 94558,c1(C(C)NCCCN(C(=O)OCC)C)cccn1Cc1ccccc1 94559,c1(NC)cccc(C(N2CC(CN3CCN(C(=O)C(C)CO)CC3)C2)=O)n1 94560,C1(NC(C(C)NC(C)=O)=O)COC2(C1)CN(C(c1cnc(C(C)(C)C)o1)=O)C2 94561,N1(C(C2CN(C)C2)=O)CCCC1C(=O)N(C)Cc1nnc(O)o1 94562,c1(C(=O)NCC2(O)CN(C(C(C)Sc3nncn3C)=O)C2)nn(C)cc1N 94563,c1(OC)ncc(C(=O)NCCOC2CN(C(=O)C(c3cccnc3)=O)C2)s1 94564,c1(CNC(C23CC(Nc4c(C)c(Br)cnc4)(C2)C3)=O)ccc(F)cc1[N+](=O)[O-] 94565,c1(NC(C)CC(C)NC(C2CCC3CC3CC2)=O)c([N+](=O)[O-])cnn1C 94566,c1(C2(N(CC(=O)O)Cc3cnc(CCCC)[nH]3)CC2)ccc(F)c(F)c1 94567,n1(CCCSC)nnnc1C(C1(N)CC1)NCc1ccccc1.C(C)(C)(C)OC=O 94568,C1(CC)CN(C(=O)CC(C(F)F)NC(=O)C(C)=C2CCC2)CCCO1 94569,c1(OC)cccn2ncc(C(=O)N(C3CN(C(=O)CN4CCC4C)CC3O)C)c12 94570,c1(OCC=CC)cc(CC(=O)NC2(CCNC(=O)CC(C)(F)F)CC2)cc(F)c1 94571,c1(C(N2CCC3CN(C(C4CCN(C)C4=O)=O)C3C2)=O)ccc2c(c1)OCCC2 94572,c1(C(=O)NC(c2ccc(F)cc2)CNC(C(C)SC)=O)ccc(F)c2c1OCC2 94573,C12(CNC(c3cn(CCC)nc3)=O)CC1CN(C(=O)CC1CCC1(F)F)C2 94574,C1(C(N2CCN(C(CNC(=O)CC(F)(F)F)=O)CC2)=O)CCc2nc(O)[nH]c2C1 94575,Cc1c(C(=O)NCC2(CC(N3CCCC3C(N)=O)=O)CC2)[nH]ccc1=O 94576,Cc1noc(C)c1C(=O)Nc1ccsc1C(=O)NC1CC1(F)F 94577,c1(OC)ncc(Br)c(=NC(=O)C2CCCC(NC(=O)CCCCCBr)C2)[nH]1 94578,CC1(C(N2CC(C(N)=O)C(c3ccccc3)C2)=O)Oc2ccccc2NC1=O 94579,N1(CC2CC(C)C2)CC2C3CCC(C2C1)N(C(c1cc(O)cc(=O)o1)=O)C3 94580,c1(NC(C2COCCN2C(C2CC2C2CC2)=O)=O)cc(F)ccc1Br 94581,N(C(=NCCc1cncnc1)NCCN1CCCC1)CC1(C)CCCCO1 94582,C1(O)(C(N(C(C)CCNC(=O)CC2(C)CCOC2)C)=O)CC2CCC1C2 94583,C1(CCNC(C(C2CCCN(C(C3C4CN(C)CC34)=O)C2)C)=O)CCCC2CC12 94584,C1(C(=O)NC2C(NC(Cc3c(C)cco3)=O)CCCC2)CN2CCN1C(C)C2 94585,C1(CCC)CN(C(c2nc(C)oc2OCC)=O)CCN1C(c1cc(=O)cc[nH]1)=O 94586,c1(C(=O)NC(C)(CNC(c2cn[nH]c2)=O)Cn2cccn2)cccc2scnc12 94587,c1(C(=O)NC2(C3CN(C(=O)C=CCO)C3)CC2)cc2cc(Br)ccc2s1 94588,c1(C(=O)NCC(CC(=O)N(C)Cc2c(C)nco2)C)ccc(F)c(F)c1 94589,c1(C(=O)NCC(=C)CCNC(=O)Cc2occc2C)ccccc1SCC 94590,C1(C(=O)NCCC2CSCCN2C(=O)C(C)N=[N+]=[N-])(CC)CC(C)(C)C1 94591,N1(C(C(C)=C(C)C)=O)CCCC12CCN(C(=O)CCCC1CC1)C2 94592,C(=O)(C(C)(C)C(=O)N1CC2C(OC)C2C1)NCCOc1c(OC)cccc1 94593,c1(C(C(=O)NCC(C2CCC2)NC(CSC(C)C)=O)(F)F)ncc(Cl)n1C 94594,c1(C(=O)NCC(CNC(CCOCC#C)=O)C)ccc(N(C)CC2CC2)cn1 94595,c1(C(=O)NC(CC)(CNC(=O)C(F)(F)COC)CC)ccc2cccnc2n1 94596,c1(N2CC3N(C(C4N(CCCC)CCCC4)=O)C3C2)nc(COC)ncc1Br 94597,C(C)(C)(CCNC(=O)Cc1cc(C(C)C)no1)NC(COCC(=O)NC)=O 94598,CC(=O)CCC(=O)NC1CC(OCC(=O)NCC(C2CC2)C2CC2)C1 94599,C1(NC(c2cc(-c3cn(C)nc3)no2)=O)CN(C(=O)CNc2nccs2)C2CC12 94600,c1(C(C(=O)NC2CC2)N(CCOC)CC)cc2n(n1)CC(C)(C)CO2 94601,C(C(C)(C)C(=O)N1CC(O)(C(C)(C)CNC(C2CCC(C)(C)O2)=O)C1)SC 94602,c1(OC)c(Cl)ccc(C(=O)NCC2CC(C)CCN2C(C23CC(OC)C2C3)=O)c1F 94603,N1(C(C(CC=C)C)=O)CC2(C1)CN(C(C1(c3ccccc3)CC1)=O)CC2CO 94604,Cc1cc(C(N2CC3CCC2C(NC(=O)C(F)C2CCOC2)C3)=O)c(Cl)cc1F 94605,c1(CC)ccc(C2(C(N3CCC(N(C(=O)COCCF)C)C3)=O)CCCC2)cc1 94606,Cc1cc(F)ccc1CN(CCOCCNCCOC(=O)C1CC1)CCN.NC=O 94607,c1(C(N2CCC(c3nncs3)C2)C(=O)NCCCSC)cccc(CO)n1 94608,Cc1ccc(C(=O)NCCNC(N2CC(CO)CC2C)=O)cn1 94609,c1(C(=O)OC)cc(NCC2(C(C)(C)O)CCOC2)cc(Cl)c1C#N 94610,c1(OC(c2nccn2C)C)ccc(NC(C2CCC(C)(C)CO2)=O)cc1Cl 94611,CCCCC(O)CC(=O)N(C(CC)CC(N1CCC2(CCCO2)C1)=O)C 94612,c1(CC)ccc(NC(C2CC(C)(NC(=O)CC(C)O)C2)=O)cc1Cl 94613,c1(C(=O)NCC2(F)CCN(C(CSCCOC)=O)C2)ccc2occ(C)c2c1 94614,N1(C(COCC)=O)CCCC2C1CCN2c1ncc(Br)c(OC)n1 94615,C(=O)(C1=CCSC1)N(C(C)(C)CC(=O)NC1(C)CCOCC1)C 94616,C1(C(=O)NCCCn2cc(CC3CCNC3=O)nn2)C2Cc3cc(Cl)ccc3C12 94617,c1(C(N(C)CC2CCCN(C(c3c(C)cn(C)n3)=O)C2)=O)cc2cccnc2s1 94618,N1(C(c2cncc(OC)c2)=O)CCCC(C)(C(N2C(C)CCC2(C)C)=O)C1 94619,C1(NC(c2nc(COC)sc2)=O)CCCC(C(NCP(C)(C)=O)=O)C1 94620,C=CC(C)(O)C(=O)N1CC(NC(=O)CCOCC)C(C(F)(F)F)C1 94621,CN1CCN(C(=O)C(C)(C)n2cnnn2)CC1CNC(=O)C(F)(F)C1(O)CCC1 94622,C=C(C)CC(C(=O)NC(c1cccc(F)c1)C)NC(=O)C(=O)NCC(F)F 94623,c1(C(=O)NCC(=O)NC2C(CNC(c3ccn(CC)n3)=O)C2)ccc(F)c(Cl)c1 94624,c1(C(C)(C)C)nc(=NC2(CNC(C3CCC4(CC3)CC(O)C4)=O)COC2)s[nH]1 94625,c1(N2CCC(CCF)CC2)nc(N2CCC3C(C2)C3(F)F)c2[nH]ccc2n1 94626,C1(OC)(CNC(C2CC2C)=O)CCN(C(c2sccc2CC#N)=O)C1 94627,c1(C(N(C(CNC(C2CCN(C(CC)=O)C2)=O)C)C)=O)cc([N+](=O)[O-])cc(C)n1 94628,C1(NC(C2CC(C(F)F)C2)=O)CN(C(c2ccc(N3CCC3)nc2)=O)CC1CO 94629,c1(N2CC(CN(C)C(c3c[nH]cc3Br)=O)C2)nc(Cl)nc2c1ncn2C 94630,c1(NCCC(CCC)C)ccc(S(=O)(=O)NCc2cc(C)nn2C)cn1 94631,c1(C(=O)Nc2c(C)n(-c3ccc(OC(F)F)cc3)nn2)cn2cc(F)ccc2n1 94632,CC1SCCN(C(=O)C(C)(C)C2CCN(C(=O)C#CC3CC3)C2)C1C 94633,CC1=C(C(=O)N2CCCCCC2C(=O)NCCC2(C)CCCC2)COCC1 94634,c1(C(N2CCN(C(C(CC)CC)=O)C(CC3CC3)C2)=O)ccc2c(c1)COCO2 94635,C(=O)(CCC(=O)N(CC(N1CCC(CC2CC2)C1)=O)CCC)NCCC 94636,Cc1cc(N)c(C)nc1C(=O)NC1CCN(C(=O)C(c2ccc(F)cn2)(F)F)C1 94637,CN1CCN(C(=O)CC2CCCCO2)C(CNC(C2C(C)(C)C2(C)C)=O)C1 94638,c1(C(=O)NCC=C2CCN(C(c3cnc(C)n3C)=O)CC2)cnn2c1N(C)CC2 94639,n1(CC(=O)NCC(CN(C(C2CCCC2O)=O)CC)(C)C)nnc2ccccc12 94640,N1(C(c2cc(-c3ccc(C)s3)[nH]n2)=O)CC2(CCCC2NC(C2CC2C#N)=O)C1 94641,c1(C(=O)NC2C(C)CN(C(=O)C(CC(F)F)C3CCC3)C2)cccc2nccn12 94642,C1(CNC(C(=Cc2ccccn2)C)=O)CN(C(=O)Cc2csnc2C)CCCO1 94643,C(CCCCCNC(=O)C(F)F)NC(=O)C(c1cccc(C(F)(F)F)n1)(F)F 94644,c1(C(=O)NCc2c(C)c(Cl)ncc2)n[nH]c2c1CN(C(C1CC1C)=O)CC2 94645,c1(C(=O)NC2(CCCNC(C(CCCOC)C)=O)CC2)cc(O)c2ccsc2c1 94646,c1(N(CCCC)C)ncnc2c1ncn2CC(C)(Cc1ccccc1)CO 94647,C1(CNC(C2CCCO2)=O)CC2CC2N1C(=O)CC1CC(n2cnnc2)C1 94648,C(=O)(CC(C)CC(C)C)N1C(C(=O)NCC2(CC)CC2)CSCC1 94649,N1(C(C(OC)OC)=O)CCN(C(=O)CCCSC)CC(CO)C1 94650,C(=O)(C(CN(C)C)C(C)C)N1CCC(N(C(=O)CNC2(C)CCCN2)CC)C1 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94669,N1(C2CN(C(=O)CC3CC3(Cl)Cl)C2)CCN(C(c2ccc(CF)cc2)=O)CC1 94670,C(=O)(C1CCCn2cnnc21)NC1C(C)CN(C(c2c(Cl)cncc2Cl)=O)C1 94671,c1(C(=O)NCC2C(CNC(=O)CCCF)C2)ccc([N+](=O)[O-])c(C(=O)CC)c1 94672,c1(C(c2n(CCOC)nnn2)NCC2(Br)CC2)nc(Br)cn1C 94673,c1(C(=O)NCC2C(CNC(C3CC(CC)OCC3)=O)C2)nc(N(C)C)nc(=N)[nH]1 94674,c1(C(=O)NC(COCC)C(=O)N2CCC(O)C2)ccc([N+](=O)[O-])[nH]1 94675,N1(C(C(C)(C2CC2)OC)=O)CCC2(CC1)CC(NC(=O)C=CC1CC1)CCO2 94676,C1(F)(C(N2CCC(CC(C)O)CC2)=O)CCN(C(c2ccsc2C#N)=O)CC1 94677,C(=O)(CCCCCF)NC(CC)CNC(=O)C=Cc1nnc(C(C)C)o1 94678,c1(C(=O)NCC(C)(C2CC2)NC(CC(CC)C)=O)cccc(-c2ccccc2)c1O 94679,C1(NC(C2=CC(C)C2)=O)CCC12CCN(C(=O)Cc1cnnn1C)CC2 94680,N1(C(C2(C)CCC(C)C2)=O)CC(C2CN(C(c3nn[nH]c3C(F)(F)F)=O)C2)C1 94681,C1(c2ccccc2)(CNC(N2CCCC2c2cncc(Br)c2)=O)CC2CCC12 94682,c1(OCC)cccc(CC(=O)NC(C)CNC(=O)CC2COC3CC2C3)n1 94683,C(CCC(C)(C)NC(c1ccc(C)nc1)=O)NC(CCCOCCOC)=O 94684,C(=O)(C1=C(Cl)CCC1)NCC(C)(C(=O)O)OC 94685,N1(C(=O)CC(F)(F)F)CC2(C1)CN(C(C1C(C3CC3)C1(F)F)=O)CCO2 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94703,CC1(C)CC2(CC(C(=O)NCC3CCCN3C(=O)Cc3cccc(F)c3F)C2)C1 94704,c1(OCC)nc(C)ccc1C(N1CC(NC(c2cnc(SC)s2)=O)C(O)C1)=O 94705,N1(C(c2ncnn2-c2ccccc2)=O)CCC2C(C1)C2(F)F 94706,c1(C(=O)Nc2c(C)nc(C(F)(F)F)cc2)cnn2ccc(CN)cc12 94707,CS(=O)(=O)CCCC(=O)NCC1(F)CCC(NC(C2CN(S(C)(=O)=O)C2)=O)C1 94708,C1(C(=O)NCC2C(C)(C)CN(C(=O)COCC(F)F)C2)COc2ccccc2O1 94709,C1(N(C(c2csc(C(=O)OC)n2)=O)CC)CCN(C(=O)C(C)CO)CC1 94710,c1(C2(C(=O)NCC3CN(C(C(=O)NC(C)C)=O)C3)CCC2)ccccc1 94711,c1(C(=O)NCC(C2CCCCN2C(C2CC2(F)F)=O)(C)C)cccc(N)c1 94712,C1(C(=O)NCc2ccc(C)cn2)CN(C(=O)C2=COCCC2)CC1(F)F 94713,C(=O)(C1=C(C)CCC1)N1C(CC=C)(C(N2CC(c3nncs3)C2)=O)CCC1 94714,C1(C(N)=O)CCC(C(=O)NCCCn2ccnc2)CC1.c12csc(n1)CC(=O)N2 94715,C1(NC(c2cc(C(F)F)no2)=O)CC2CN(C(=O)Cn3nccn3)CCN2C1=O 94716,CCCCCCC(F)C(=O)NCC(CC)NC(c1nc(C)sc1C)=O 94717,CC(CC(C)(C)C)C(=O)N(CCCN(C)C(c1cc(C(F)F)no1)=O)C 94718,N1(c2cc(OCC)ncn2)CCC2(CCOC2)C(CNC(=O)CCC2(C)CC2)C1 94719,N1(C(CCNC(=O)NC)=O)CC2(COC(CNC(c3cc(Br)no3)=O)C2)C1 94720,c1(OC)ncc(NCc2ccc(-c3ccccc3OC(F)F)s2)cc1Br 94721,O=C1CCCCC(C(=O)NCCC(O)C(=O)N2CCCC2C2CCOC2)C1 94722,N1(C(C(C)OCC(F)(F)F)=O)C2CCC1C(CNC(c1ccccc1)=O)C2 94723,c1(C(=O)NCCC2(OC)CN(C(c3scc(OC)c3)=O)C2)cc(C)cc(O)n1 94724,C1(C)(C(=O)NCCCCC)CCCN(C(c2cccc(OC)c2O)=O)C1 94725,C1(CNC(=O)Cc2cnoc2)CCCC1C(=O)NC1C2CCCC12 94726,c1(OCC(=O)OC)cccc(CC(C)NC(c2ccccc2-n2cccc2)=O)c1 94727,c1(C(=O)NC(C2CCCC2)CNC(CC(=O)NCC#C)=O)nnn2c1COCC2 94728,N1(C(C(C)OCC)=O)CCC2(CC1)COC(CNC(=O)Cc1cncc(C)c1)C2 94729,C1(NC(CSCC(=O)OC)=O)CC2CC1N(C(=O)CCOc1cccc(C)c1)C2 94730,C1(CC)CCN(C(C2CCS(=O)(=O)C2)=O)C1CNC(c1ccc(SC)o1)=O 94731,O=C(CC1OCc2ccccc21)NC1CCCN(C(c2ccns2)=O)CC1 94732,c1(OC)ccc(O)cc1NC(=O)C(C)C(C)NC(C1(C(=O)N(C)C)CCC1)=O 94733,c1(CCC)ccccc1C(=O)NCC(O)CCNC(=O)CCC1CCCCO1 94734,c1(N2CCC(NC(C(C)CSC(F)(F)F)=O)C2)nnc2c(c1C#N)CCCC2 94735,c1(C(=O)NCCC(=C)CNC(c2cc(O)n(CC)n2)=O)cc[nH]c(=NCC)c1 94736,C1(NC(C2CCC(=O)N2)=O)COC2C(NC(c3cnn(C4CC4)c3)=O)COC12 94737,c1(C(=O)NC2CCN(C(C(n3ncc(C)c3)C)=O)C2)ccccc1CO 94738,N1(C(CN2CC(=O)NCC2)=O)CCC2(CCCC2NC(c2ccccc2)=O)CC1 94739,Cc1nc(O)c(Br)cc1C(=O)NC1(CO)CN(C(=O)C(Cl)=CCl)C1 94740,c1(C(=O)NCC(C(C)C)NC(c2ccc(C(O)CF)cc2)=O)cc(Cl)n(C)n1 94741,c1(C(C)=O)ccccc1C(=O)N(C)CC1CCCN1C(=O)CC12COCC(C1)C2 94742,C(CCCC)(CC(=O)NC(CO)C(C)(C)CO)NC(CCCC#C)=O 94743,C1(N(CC(=O)NCc2cocn2)C(=O)C2CC2)CCCC12CCNCC2 94744,c1(C(N2CCC(C3CC3)C2CNC(C2(CF)CC2)=O)=O)ccc([N+](=O)[O-])cc1Cl 94745,C(CC1c2ccccc2CCN1C(=O)COC1(C)CCC1)NC(C(C)C)=O 94746,C12(C(N(C3CCN(C(=O)Cc4cc(Cl)cs4)C3)C)=O)CC3CC(C1)CC(O)(C3)C2 94747,Cc1nc2c(C(N3CC(NC(c4cc(CO)[nH]n4)=O)CC3C)=O)ccnc2[nH]1 94748,c1(OC)cnc(F)cc1C(N1CC2CCC1C2NC(=O)Cc1ccc(Cl)cn1)=O 94749,N1(C(C(CCC#C)O)=O)CC2CCN(C(c3cccc(CC)c3)=O)CC2C1 94750,c1(C(=O)NCC(C)N(C(=O)C=Cc2cscn2)CC)cnc(C2CC2)nc1 94751,C1(C)(C(=O)Nc2sc(Cc3ccc(C)cc3)c(C)n2)CCCCC1C 94752,CC(C)C(CNC(=O)C(c1cncnc1)C)C(=O)NCc1ccc(C#N)cc1 94753,c1(C(=O)NCCN(C(C2COC3(C)CC2C3)=O)CC)c(C)cccc1C 94754,C1(NC(c2n(C(C)C)ncc2F)=O)CC(O)CN(C(C2CCN(C)CC2)=O)C1 94755,c1(C(N2CC(OC)C(NC(c3occc3C)=O)C2)=O)ccnc2cc(F)cnc12 94756,CN1CCCC2CN(Cc3cc(N4CCCC4)nc(F)c3)CCC12 94757,c1(C(N2CC(n3cc(C(CC(C)C)O)nn3)C2)=O)ccc(Cl)c(F)c1 94758,N1(C(c2c(C)cns2)=O)CCC2CCC(NC(c3cc4ncccc4s3)=O)C1C2 94759,CC(C)C(F)C(=O)NCC1(F)CC(Nc2ncccc2C(=O)C(F)(F)F)C1 94760,c1(C(N(C2CCN(C(C34CC(C)(CCO3)C4)=O)CC2)CC)=O)cc(=O)cc(C)[nH]1 94761,c1(CN(C(=O)Cc2cc[nH]n2)C)cnn2c1CN(C(C1CCC(C)(C)C1)=O)CC2 94762,C1(NC(CC2CN(C(C)=O)C2)=O)CC2(CCN(C(c3ccc(C)c(Cl)c3F)=O)C2)C1 94763,N1(CC(=O)N(C(C)(C)C)CCO)CC(O)CC1c1ccc(Br)cc1 94764,c1(CC)cc(C(=O)N(CC(O)CNC(c2cnc(C)n2C(F)F)=O)C)cc(Cl)c1 94765,C1(NC(C(=O)NC2CC2)=O)CC2CCC(C1)N2C(c1ccnc(O)c1)=O 94766,c1(C(=O)NC(C2CCN(C(=O)CC3CCC3)C2)C)cscc1S(C)(=O)=O 94767,Cc1onc(C(=O)NC(CNC(=O)CC2CC(F)C2)CC(C)C)c1[N+](=O)[O-] 94768,N(C(=NCCc1ccc(Br)cc1)NCc1cnc(C)cn1)C(CC)C 94769,C(=O)(C(C(C)(C)C)NC(C)=O)N1CC(c2cn(CCC=C)nn2)C(O)C1 94770,N1(C(C=CC)=O)CCC(NC(c2ccc(N3CCCC3)nn2)=O)C(CC)C1 94771,C1(CCNC(C2(CC)COC2)=O)CN(C(c2ccc(-c3cccs3)o2)=O)CCO1 94772,c1(C(=O)NCC2(C(C)NC(C3N(CC)CCOC3)=O)CC2)ccc([N+](=O)[O-])cc1 94773,CN1CC(CCNC(C2CCCC2CNC(=O)C=Cc2cocn2)=O)CC1=O 94774,c1(NC(CCN(C(=O)C(F)C2CCOC2)C)=O)cccc2cccnc12 94775,c1(C(NOCC(=O)N(C)Cc2cccnc2O)=O)cccc2[nH]ccc12 94776,C1(C(=O)NC(C(=O)N(CC)CC)C)CC(NC(C2CC2(C)C(F)F)=O)C1(C)C 94777,c1(C(N(CCC(C(C)C)NC(COC(C)C)=O)C)=O)cc2n(n1)CCCC2 94778,c1(C(=O)NC2C(CNC(C3(CC=C)CC3)=O)C2)c[nH]c2ccc(Cl)cc12 94779,CC1CC(O)CN1C(=O)NC(C1CC(F)(F)C1)C(F)F 94780,N1(C(CCC=C=C)=O)CC2(CO)CC1(C(=O)NCCc1ccccc1F)C2 94781,c1(CNC(C(Cc2cc(C)c(O)cc2)N)=O)cnn2c1CCCC2 94782,Cc1ccc2cccc(C(=O)N(C3CN(C(c4cnc(Cl)cn4)=O)C3)C)c2n1 94783,Cc1sc2ncc(C(=O)NCC3(NC(c4cc(Br)co4)=O)CCC3)n2c1C 94784,CS(=O)(=O)c1ccnc(NC2C3CN(C(c4cc(Cl)on4)=O)CC23)n1 94785,C(=O)(C1=CCOCC1)NCCC(C)(C)NC(c1cccn(C2CCC2)c1=O)=O 94786,N1(C(c2c(C)ncn2C)=O)CC=C(CNC(=O)C(C)OCCC(C)C)CC1 94787,C(=O)(C(C(=O)N1CC2CC1C2NC(=O)C(F)C(C)(C)O)C(C)C)OCC 94788,C(=O)(C1=C(Cl)CC1)NC1CC(C)(CNC(C2(c3ccno3)CCC2)=O)C1 94789,CC1CCCC1N(C)C(C1(CCNC(=O)Cc2ccsc2)CCC1)=O 94790,C1(NC(C(COC)(C)OC)=O)CCCCCN(C(c2ccccc2Cl)=O)C1 94791,C(CCC(C)C)(C(=O)Nc1ccc(N(C)C)cc1)NC(C(CCC)CC)=O 94792,N1(S(CC)(=O)=O)CCC2(CC1)CC(C)N(C(C1CC1C(=O)OC(C)(C)C)=O)C2 94793,N1(C(c2nc(CC)sc2)=O)CCC2(CCC2)C(NC(=O)C(C)n2cccn2)C1 94794,C(C(C)C(=O)NN(C)C(C1C=CC1C(=O)OC)=O)OC.C12(CC1)CC2 94795,N1(C(C(CCCNC(c2n(C=C)ncc2)=O)(C)C)=O)CC(C)OCC(C)(C)C1 94796,N1(C(c2c(C)nns2)=O)C2CCC1C(c1cn(CC(c3ccccc3)O)nn1)C2 94797,Cc1cc(C(=O)NCC(C)(C)CNC(c2ccc(F)c(C)c2)=O)c(C)c(O)c1 94798,c1(SC)ccc(C(=O)NC(C)(C)CNC(=O)CO)cc1.C1(CN)CC1 94799,c1(C(=O)NCCN(C(=O)C(C(C)C)n2cc(Br)cn2)CC)cn(C)nc1Cl 94800,c1(C(=O)NCC(C)CN(C(=O)C(O)C2CCCC2)C)cc(OCC(F)F)ccn1 94801,N1(C(C2(F)CCN(C(c3cc(COC)on3)=O)CC2)=O)CCCC2(CCC2)C1 94802,C(=O)(C(C)CC(C)(F)F)N(C)CC1(O)CN(C(c2c(OC)c(Cl)ccc2)=O)C1 94803,C1(NC(C(CCOC)C)=O)CCC2(CC1)CN(C(=O)CCF)C2 94804,c1(N(C)C)nc(F)ccc1CNc1ccc(C(=O)Nc2ncc(Br)cc2Cl)nc1 94805,C1(SC(F)(F)F)CCN(C(=NCCc2ccc3c(c2)COCC3)NC2CCC2)C1 94806,C=Cn1nccc1C(=O)NCC(CC(=O)NCCN(CCCF)C)C1CCC1 94807,c1(C(=O)NCCC(CNC(CC2N(CC)CCC2)=O)O)cc(O)n(CC)n1 94808,c1(C(=O)NC(CC=C)CNC(c2c(C)cccc2C)=O)n[nH]c2c1CC1CC21 94809,C(=O)(C(C)CN(C)C)N(CCC(=O)NC1(C(=O)NCCC)CC1)C 94810,c1(NCC2C(CCC)C2)cc(=NC2CCCN(CCC)C2)[nH]c(C(F)(F)F)n1 94811,CCC(C)(C)C(=O)N1CC(CC(C)(C)CNC(c2nocc2Cl)=O)C1 94812,c1(C(=O)NCCC(C)N(C)C(c2ncc(Cl)cc2Cl)=O)cnn2c1OCC2 94813,N1(C(C(C)=CC2CC2)=O)CC2CC(C1)CN(C(=O)C(O)(C1CC1)C1CC1)C2 94814,CC1CN2CCN1CC2C(=O)NC1CC(C)(NC(c2ccncc2N)=O)C1 94815,c1(-c2cnc(SC)nc2)cccc2c1CCN(S(=O)(=O)CCCCCl)C2 94816,C1(C(=O)NCC(C)(C)NC(C(C)SC)=O)CCC(=O)N(C)C1 94817,CC1CCC(CNC(C2CC(O)(C(F)(F)F)C2)=O)N(C(=O)C=Cc2ccoc2)C1 94818,CC1CN(C(C2C3CCC(C3)N2C(c2cc(Cl)cs2)=O)=O)CC(=O)N1C 94819,C(=O)(CC(C(C)(C)C)NC(=O)CC1CC2CC2C1)NCC12N(C)CC(C1)C2 94820,c1(CCNC(C(C)NC(c2ccc(Cl)cc2)=O)=O)c[nH]c2cnc(Cl)cc12 94821,C(c1ccccc1)=CC(=O)NCCCOCCNC(C(OC)OC)=O 94822,C1(C(=O)NCCCN(C(C=C(C)Cl)=O)CC2CCCC2)CCC2(CC2)C1 94823,C(=O)(C(C)CC(=O)N1CCC(n2cc(-c3cc(CO)ccc3C)nn2)C1)OC 94824,C(=O)(C(C#N)C(C)(C)C)N(CCCN(C)C(C1CCCC1F)=O)C 94825,C1(C(=O)NCC2(C(N(C)Cc3cc(C)n(C)n3)=O)CCCO2)CCCC1C1CC1 94826,CC(C)(C#CC(=O)NC1CC2OC(=O)CC12)CNC(C1(COCC2CC2)CC1)=O 94827,C1(C2CC2)(CNC(CCCCCC)=O)CCN(C(=O)C(C)(C)C(O)CC)C1 94828,c1(C(C(=O)NCC(C)CNC(C2(C)CC=CC2)=O)=O)c[nH]c2ccccc12 94829,Cc1cccc(C(N2CCC(NC(C3CCC(C)(C)CO3)=O)C2)=O)c1C(F)(F)F 94830,CC1(NC(=O)C(O)CC(F)F)CCN(C(=O)Cn2ccc(C3CC3)n2)CC1 94831,O=C(CCc1ccccc1)C(=O)NCC1CCCN1C(=O)Cc1nccs1 94832,c1(OCC)nc(NCc2c(C(=O)NC(C)(C)C)cccc2)ncc1Br 94833,CCCC(C)(C)C(=O)NC(Cc1ccccc1)CCNC(c1ccc(Cl)nc1O)=O 94834,C(=O)(CCCC(C)C)N1C(C2CCN(C(Cn3ncc(C)c3)=O)C2)CCCC1 94835,C1(C(=O)NCC2(NC(CC3(C)CCCCC3)=O)CCC2)C2Cc3ccccc3C12 94836,CC(C)(C)C(C)(C)C(=O)NC1CCN(C(c2cnc[nH]2)=O)C(C2CC2)C1 94837,N1(C(C(C)N(C(c2cc(C3CC3)[nH]n2)=O)C2CC2)=O)CCCC(C2CCC2)C1 94838,c1(OC(C(N2CC(C)(NC(c3c(NC)cncc3)=O)C2)=O)C)ccc(C#N)cc1 94839,C1(C(F)(F)F)(C(=O)NC)CCN(Cc2ccn(C)n2)C1 94840,C#Cc1nccnc1NC(C1CC12CCN(C(c1c(OC)cccc1F)=O)C2)=O 94841,c1(C(N(C2CN(C(C(CCC)N(C)C)=O)CC23CC3)C)=O)nnn2c1CCCC2 94842,C1(CNC(C(N2CCS(=O)CC2)(C)C)=O)CN(C(=O)C2=COCC2)C2(CCC2)C1 94843,N1(C(C2C(C(C)(F)F)C2)=O)CC2CC(C1)N(C(c1nn(C(C)C)c(C3CC3)c1)=O)C2 94844,C1(CCC)CN(C(=O)Cc2c(C)noc2C)CC1C(=O)NCC1CCC=CCC1 94845,N1(C(CN2C(=O)CCCC2)=O)CCc2onc(C(=O)N=c3cncc(Cl)[nH]3)c2C1 94846,N1(C(c2c(C)nn[nH]2)=O)CCC(NC(C2CCN(C(=O)N(C)C)C2)=O)C12CC2 94847,N1(C(C2C(OCC)C2)=O)CCCCC(CNC(=O)C(c2cc(Cl)cc(Cl)c2)O)C1 94848,C(=O)(C1CSc2ccccc21)NC1CCN(C(c2c(N)cc(F)c(Cl)c2)=O)C1 94849,C(=O)(C1CC(=O)Nc2cc(F)ccc21)N(C)CCNC(c1nscc1Br)=O 94850,N(C(=NCC(C)(C)C1(O)CCC1)N1CCC(NC(=O)CC(F)(F)F)C1)C(CC)C 94851,O=C(C1=CC2CCCCCC12)NCC1CCN(C(c2cnc(Cl)[nH]2)=O)C1 94852,c1(C(N2C(C(=O)NCC(CC)C)CC3CC32)=O)cc(C)cc(O)n1 94853,N1(C(CC2CC(C)N(C(=O)CCCC(C)(C)C)C2)=O)CCOCC(C)(C)C1 94854,c1(C(=O)NC2CCC(N(C(C3C(C=C)CC3)=O)C)CC2)cc(Br)ccc1N 94855,C(=O)(C(CC(C)C)ONC(=O)C(F)=C1CCC1)N1CCC(CC=C)C1 94856,N1(C(CCCCC=C)=O)CC2CCN(C(c3ccc(=O)n(C)n3)=O)C(C2)C1 94857,CCC(CN=C(NC(C)C1CC1)NC1CCOCC1)Oc1cccc(C)c1 94858,C1(C(=O)NC(COCC)C(=O)N2CC(N3CCCOCC3)C2)CCC(F)(F)C1 94859,c1(C(N(c2ccc(OC)cc2)C)=O)cc(N2CCOCC2)cc(F)c1 94860,C1(C(C)C)C(C(=O)NCC(C)(C)C)CCN1C(=O)CCC1CCC(=O)C1 94861,N1(C(C(C(=C)Cl)(C)C)=O)C2CCCC1CC(NC(c1cscc1C(F)(F)F)=O)C2 94862,c1(C(=O)NC(C)(C)CNC(=O)COCCCF)cc2c(s1)COCC2 94863,C1(N=[N+]=[N-])(C(N(C)CC2(C#N)CCC2)=O)CCN(C(=O)CC(F)(F)C(F)F)C1 94864,C1(NC(=O)CCCc2cncs2)CC2CC1N(C(=O)CCCn1cccn1)C2 94865,c1(C(N(CCNC(Cc2cn(C)nn2)=O)C2CC2)=O)noc2c1COCC2 94866,c1(C(N(C2CCN(C(C3CCC4(CC4)C3)=O)C2)CCO)=O)ccc(F)cc1O 94867,c1(C(=O)NCC2CC3CC3N2C(c2cccc(C(F)F)c2)=O)occ2c1CCC2 94868,C(=O)(N1Cc2ccccc2CO1)c1nn(C)c(C(=O)O)c1Br 94869,N1(C(CN(CCC)C)=O)CCC2(CC1)CC(CNC(=O)Cc1csc(Cl)c1)C2 94870,N(C(=NCC1CCSC1)NCc1ccco1)Cc1c(COC)noc1 94871,N1(C(C(C)NC(=O)NC)=O)CCCC(N(C)C(c2csc(CC(C)C)n2)=O)C1 94872,N1(C(c2cnc(OC)nc2)=O)CCN(C(=O)CC(C)C)CC1C(C)C 94873,c1(SC)cccc(F)c1CNC(=NCC1C2CCC(F)(F)C12)NCC1CCCO1 94874,c1(C(=O)NC2CCN(C(C=Cc3ccc(OC)cn3)=O)C2)cc(C#N)c(C)cn1 94875,N1(C(c2cc(CC)[nH]n2)=O)CCN(C(=O)Cc2nc(=N)[nH][nH]2)C(C2CCC2)C1 94876,C=CCC(CC(C)C)C(=O)NCC(CC1CC1)C(=O)N(C)Cc1cocn1 94877,C(=O)(CCC(=O)NC(C(=O)NCCCc1cccnc1)C1CCCO1)NC 94878,CC1CCN(C(c2ccc(C(=O)NCc3cccc(F)c3)cc2)=O)CC1(C)O 94879,Cc1c(Br)cnn1CC(=O)NCCNC(c1cc(Cl)n(C)n1)=O 94880,C1(C(=O)NCC2(CO)C(C=C)C2)N(C(=O)C2=C(Cl)CCOC2)CC12CCCC2 94881,C12(CNCC(=O)NC3CCSC3=O)CCC(O)(CC1)CC2 94882,C12(C(=O)NC3CN(C(CS(=O)(=O)NC)=O)CC3C)CC(C)(C1)OC2C 94883,C1(C)(CNC(CNC(CC)=O)=O)CN(C(=O)CC(C)NC(N)=O)C(C)(C)C1 94884,N1(C(COCCOC)=O)CCCC1(C)CNC(=O)CCc1n[nH]c(=N)s1 94885,CCCC(C)(O)CC(=O)NC1C2CC(NC(c3cc(OC)nn3C)=O)CC12 94886,c1(C(=O)NCC(F)CNC(=O)C(F)F)ncnc2c1CCC2 94887,C1(C(=O)NC2C(CC)N(C(c3cc[nH]n3)=O)CC2)CCCC2(CCOCC2)O1 94888,c1(OC)ccc2nc(C)c(C(=O)NCC(C)CNC(c3c(C)ccn3C)=O)n2n1 94889,CC1CN(N2Cc3ccc([N+](=O)[O-])cc3C2)CC(C)N1C1CC1 94890,N1(C(c2cnc(C(C)C)o2)=O)CCN(C(=O)COC2CC=CC2)CC(C)C1 94891,C1(NC(=O)CC2CCCCO2)CCCC(C(N2C3COCC2C3)=O)C1 94892,C(=O)(C(C)(C)CS(N)(=O)=O)NCC(CC)NC(c1c(Cl)ccc(Cl)c1F)=O 94893,CC1(C(=O)OCC2CCS(=O)(=O)C2)CC2(C1)CC(F)(F)C2 94894,N1(C(C=CCN(C)C)=O)CCC(C2CCCN(C(c3ccn(O)c(=O)c3)=O)C2)C1 94895,c1(C(C(CC)NC(=O)C(F)CC2CN(C(=O)OC(C)(C)C)C2)=O)ccc(F)cc1F 94896,c1(C(N(CCNC(COCCC=C)=O)CCC)=O)oc(-c2ccccc2)nc1C 94897,c1(C(N(CCCCCNC(c2cc(SC)c(C)o2)=O)C)=O)c(C)nc(C)n1O 94898,C1(O)(CC(=O)NC(CC)CNC(=O)CC23CCC(CC2)C3)CCCN(C)C1 94899,CCC(CNC(=O)CC1CCN(C(=O)COC2CCCCC2)CC1)C(C)C 94900,N1(C(=O)Nc2c(CC)n(C)nc2)c2ccc(Cl)cc2OCC1C 94901,CC(C(=O)N(C1CCN(C(=O)COC2CCCOC2)CC1)C)S(C)(=O)=O 94902,c1(C(=O)Nc2ccc(-c3csnn3)cc2)cccc(OCc2nccs2)c1 94903,CC1CCc2c(sc3ncnc(N4CCCCC(NC(=O)CC=C(Cl)Cl)C4)c23)C1 94904,N1(C(C(C)NC(C2CCC2)=O)=O)CCCCC(NC(C2CCC3CC3CC2)=O)C1 94905,C1(OC)CC(CNC(C2CC(F)C2)=O)(NC(=O)C=C2CCCCC2)C1 94906,n1(CC=C)ccnc1C(=O)NC(C)CCCNC(c1n[nH]cc1C)=O 94907,c1(OC)nc(C)ccc1C(=O)NC(CO)C(C)NC(=O)CCC1C(=O)NN=C1C 94908,N1(C(c2c(C)nccc2)=O)CCC(C)C(CNC(C23CCC(CC2F)C3)=O)C1 94909,N(C1c2ccc(Br)cc2CC1(F)F)CCc1ccc(OC)cc1Cl 94910,c1(C(=O)NCC(CNC(C(C=C)(C)O)=O)CO)cc(OC)cnc1F 94911,C(C)(CCN=C(NCc1ccnn1C)N1CCCC(O)CC1)OC 94912,CCC(C)CCCC(=O)N(C)CC1CCN(C(=O)Cc2cc(C)no2)C1 94913,CC1CCN(C(C2CCCO2)=O)CC1CNC(c1ocnc1C1CC1)=O 94914,c1(C(=O)NCCNC(C2CN(C(C(CC)O)=O)C2)=O)oc(CO)cc1C 94915,C1(NC(C=CC(CC)=CC)=O)CC2CC1N(C(=O)C(CC)Oc1ccccc1)C2 94916,C(=O)(C(CC(=C)C)NC(=O)C(F)F)N(C(CC#C)C)C 94917,O=C(O)CC(Cc1cccc(F)c1)NC(c1ccnn1-c1ccncc1)=O 94918,C1(c2cn(C3COC(=O)O3)nn2)(NC(=O)Cc2ccc(F)nc2)CCOCC1 94919,C1(O)(CC(=O)NCCN(CCC)C(C2(c3ccn(C)n3)CC2)=O)CCCCC1 94920,C12(C(=O)NCC3CCCN(CC)C3)CCCC1CCN2C(=O)C(O)CCC(C)C 94921,C(=O)(C1=NOC2(CCC2)C1)NC1CCCC(C(N(C)CC2CN(C)C2)=O)CC1 94922,c1(OC)cccc(OCC(=O)N(CCCCCNC(C2(C)COC(=O)C2)=O)C)c1 94923,C1(NC(CCn2ccc(C)n2)=O)CC2CC(NC(C3CCCC34CC4)=O)CC2C1 94924,N1(C(=O)Nc2ccc(C(F)(F)F)cc2Cl)CC(C2CCOCC2)C1 94925,C#Cc1cc(C(=O)N(CCC(N2CC(C)(C)CCC2CC)=O)CCO)ccc1C 94926,C1(NC(CSC(C)C)=O)CCCC(CF)C1.C12CN(C1)CCNC2=O 94927,CCC(CC(=O)NC(Cc1ccco1)C(=O)NCCN1CCC(CO)C1)C(C)C 94928,CCC(COC)(CC)C(=O)N1CC(=O)CC1C(=O)NC(c1nccs1)C 94929,C(=O)(CCC1=CCCCC1)NCC1CN(C(CC(CC)(C)C)=O)C2(C1)CCC2 94930,C1(C2(O)CCN(C(C3CCC3)=O)CC2)(NC(c2ccc3c(n2)OCCO3)=O)CC1 94931,CC1CC(C(=O)NCc2nocc2C(N2CC(C)(CCO)C2)=O)CC(=O)N1 94932,N1(C(c2c(C#N)ccnc2)=O)CCC2(CC1)OCCC2NC(=O)Cn1nccn1 94933,CN1N=C(CC(=O)N2CCCC(n3cc(-c4cnn(CCl)c4)nn3)CC2)CC1=O 94934,C(=O)(C1CCc2ccc(Cl)nc21)NCC1(NC(=O)C=CCO)CCC1 94935,N1(C(CNC(C)=O)=O)CC(NC(=O)C2=NOC(C)(C)C2)C2(CCCC2)C1 94936,C1(C(=O)NCC2C(N(C)C)C2)(NC(C)=O)CCC1.C12CN(C1)C2=O 94937,C1(C(N(CC)Cc2ccoc2)=O)(CC)CN(C(C2CCCC2F)=O)C1 94938,c1(SC)ncc(C(N2CCC(NC(C3CC=CC3)=O)C(O)C2)=O)c(O)n1 94939,Cc1cc(=NCC=CBr)[nH]c(N(C)Cc2ccc(F)c(C)c2)n1 94940,C12(C(=O)NCCC(C)N(C)C(c3ncoc3C3CC3)=O)CCC(C)(CO1)C2 94941,N1(C(C(COC)(C)O)=O)CCC(NC(c2cccc(COC(F)F)c2)=O)C(C)C1 94942,c1(CNC2CCCC(C(=O)OCC)C2)c[nH]c2ccncc12 94943,C1(C(=O)Nc2ccc(Br)nc2Br)CCC2(CN(C(c3csc(Br)c3)=O)C2)O1 94944,C(CC(C(=O)NCC(N1CCCCC1)C)NC(=O)CCC(=O)C1CC1)SC 94945,C1(C(N2CC(C(C)NC(=O)C(C)n3cncn3)C2)=O)(COC)CCCO1 94946,C1(CNC(c2cc(C(C)C)[nH]n2)=O)CN(C(c2cc(Cl)c[nH]2)=O)CC1C 94947,c1(OCC(=O)NC2CC(NC(CC(C)OC)=O)C2(C)C)cc(Br)ccc1F 94948,C1(NC(c2cc[nH]n2)=O)(CO)CCN(Cc2cccc(Br)c2F)CC1 94949,C(=O)(C(C)(COC(C)=O)OC)NCC1C(NC(c2ccn(CCCC)n2)=O)CCC1 94950,N1(C(C2(CC(=O)OC)CC2)=O)CCC(C(C)C(=O)N(C)Cc2nncn2C)C1 94951,N1(CCOC)CC(C(=O)NC(C)(CNC(c2cc[nH]c2)=O)C(C)C)CC1=O 94952,Cc1cc([N+](=O)[O-])c2nonc2c1NC(C)CCN1CCCC1 94953,CC1CN(Cc2cccc(O)n2)CCN1C(=O)CN1C(C)CCC1C 94954,C1(CNC(Cc2cncc(C)c2)=O)CCC(C)(C)CN1C(=O)C(C)NS(C)(=O)=O 94955,CN1CCC(N2CCN(C(C3CCN3Cc3ccncc3C#N)=O)CC2)CC1 94956,C1(C(N2CC(N(C)C(c3cnc(S)[nH]3)=O)C3(C2)CC3)=O)Cc2n[nH]cc2C(=O)N1 94957,N1(C(=O)C(O)c2cnc[nH]2)CC2CCCC(C1)N2C(=O)C(O)c1ccsc1 94958,C1(C)(C(=O)OC)C=CCN1C(=O)C(F)C1CC(NC(C2CC(O)C(F)C2)=O)C1 94959,CC1CCN(C(=O)Cn2cc(CO)nn2)CCN1C(C12COCC1C2)=O 94960,N1(CCN(C(C(=O)NCc2ccccc2)=O)CC2CC2)CCCOC1=O 94961,C1(F)(CNC(CCCC)=O)CCC(NC(c2ccc(N(CC(C)C)C)nc2)=O)C1 94962,c1(CCC)ccc(CN(C2COCCC2CO)CC)cc1C 94963,C(c1ccc(O)cc1)=CC(N1CCCC(C(C)NC(c2cc(Br)cs2)=O)C1)=O 94964,C1(NC(C(CCCC)C)=O)CCCCCN(C(=O)CCc2cnccn2)C1 94965,C1(C(=O)NCC(CN(C)C)O)CC2(CC2)CN1C(=O)CNC(N)=O 94966,C12(C(N(CCNC(c3c(C)nc(N)cn3)=O)C)=O)CC1COC21CCC1 94967,c1(OC)c(Cl)cc(C(=O)NCC(C)(C2CC2)NC(=O)C=CC(C)(C)C)nc1Cl 94968,N1(C(C(C)NS(C)(=O)=O)=O)CCN(C(c2cccc(F)c2)=O)CC12CCC2 94969,c1(CC)cccc(C(=O)NC(C)(C)CCCNC(C2CNC(=O)C2)=O)c1N 94970,C(C(C)(C)C(=O)N1CCCC(C(N)=O)C1)NC(CC(OCC)OCC)=O 94971,C1(CN(C)C(c2ncccc2F)=O)CCN(C(c2ccn(CC(F)F)n2)=O)CC1 94972,c1(OC)ccc2c(=NCC3CSC3)[nH]c(=NCC3CC(F)(F)C3)[nH]c2c1 94973,N1(C(C(CNC(Cc2c(C)occ2)=O)O)=O)CCCC1(C)CCCO 94974,C1(CC(=O)N(c2cccc(I)n2)C)CC2CC1N(C(=O)OC(C)(C)C)C2 94975,C1(CN(C2(C)CNC2)C)CN(C(=O)OC(C)(C)C)CC1CN(C)C 94976,c1(C(N2CC(F)(CNC(C3C(C=C)C3)=O)C2)=O)oc(C2CCC2)nc1C 94977,c1(OC)ncc(C(N2CCCCC2CCNC(=O)C(O)C2CC2)=O)cc1F 94978,c1(C(N(CC(C)NC(=O)CCSCC(N)=O)CC)=O)cc(C(F)(F)F)ncc1F 94979,c1(CC(=O)NC2CCN(C(=O)CCCc3cccs3)C2)ccc(O)nc1 94980,c1(CC(C)Nc2nccc(N3CCN(C(C)=O)CC3)n2)sc2ccccc2c1C 94981,c1(C(N(C2CC(NC(C3C(C)CCC3)=O)C2)C)=O)ccnc2c1ccn2C 94982,c1(OC)ccc(C(=O)NCC2CN(C(=O)C(C)OC3COC3)CC2C)cc1O 94983,N1(C(C(C)OCC)=O)CCN(C(=O)CCc2nc3ncccn3n2)CCC1C 94984,c1(COCC)nc(C(=O)NC(C)CC(C)NC(c2cc(CN(C)C)on2)=O)cs1 94985,Cn1cc(C(O)C(=O)NCC2CCC2NC(=O)CSc2ccncc2)cn1 94986,C(=O)(C(O)C(F)(F)F)N(C)CCOCCN(C)C(C1CCC1C(C)(C)C)=O 94987,N1(C(C)C)CCN(C(=O)CCn2cc(CN3CCOC3=O)nn2)CC1C 94988,c1(C(N2CC3C(NC(c4onc(CC)c4C)=O)(C3)C2)=O)ccc(Br)nc1N 94989,C1(c2ccc(-c3ccccn3)cc2)(OC)CCN(C(=O)CCS(N)(=O)=O)CC1.c1(O)nn(C)nc1Br 94990,N1(Cc2ccc(OC)cc2)C2CCC(C2)C1C(N1CCOC(CN(C)C)C1)=O 94991,CCCCCC(O)C(=O)NC1COCC1CNC(=O)CCc1cn(C)nn1 94992,c1(C(C)C(=O)OCCn2cc(I)nn2)ccc(F)cc1 94993,C1(CC(=O)N(CCCNC(=O)CC(C)c2ccncc2)CC)CCC(=O)N1C 94994,c1(C(=O)NCC(C)NC(CCOCC(C)C)=O)ncccc1C1CC1 94995,C(=O)(CS(C)(=O)=O)NC1CCN(CCCNC(C(C)NC(=O)NC)=O)C1 94996,N1(C(C(F)=CCC)=O)CCC(C2CC2)C1C(N1CC(C)C(C)C1C)=O 94997,N(C1CCCn2ccnc21)C(C(N1CCC(Oc2ccc(C)nc2)C1)=O)=O 94998,c1(NC(C2C(NC(=O)Cc3cccs3)C2)=O)c(Cl)cnnc1Cl 94999,N1(C(C=C(CC)C)=O)CC2(CCCC2NC(c2cc(F)c(C(F)F)c(F)c2)=O)C1 95000,CC1CC2(CCN(C(C3(C(F)(F)F)CC3)=O)CC2)CN1C(C1CC12CCCC2)=O 95001,c1(-n2c(-c3sccc3Br)nc(CC(C)OC)n2)cccc2c1CCCC2 95002,C1(NC(CCN(C)CCO)=O)CN(C(=O)COC(F)F)C2(CCCCCC2)C1 95003,Cc1ncc(CC(N2CCCC2C(C)NC(C2(n3cccn3)CC2)=O)=O)o1 95004,N1(C(C2CCn3c(C)ncc3C2)=O)CCOC2(CCN(C(=O)C(C)CF)CC2)C1 95005,CC(C(=O)NC1CCC12CN(C(c1ccc(-n3cccn3)nc1)=O)C2)S(C)(=O)=O 95006,N1(C(C(CCCC=C)NC(C2C=CC2C(=O)OC)=O)=O)CCC(C2=NOCC2)C1 95007,N1(C(c2ccc(C(N)=O)cc2)=O)CC2CC(NC(c3cc(Cl)c[nH]3)=O)C2C1 95008,C(=O)(CS(=O)(=O)CCC(F)(F)F)N1C(C)CN(C(=O)CCn2ccnc2)CCC1 95009,C1(O)(CC=CC=CC)CCN(C(=O)C(C)(C)N)CC1 95010,C1(NC(=O)CC2(O)CCCC2)CCCN(C(=O)CC2CCCC(C3CC3)O2)C1 95011,C12(CCN(CC(C)(C)CC3CC3)C(c3cc(C(C)C)[nH]n3)=O)CC1COC2(C)C 95012,c1(C(=O)NCCC(C)NC(C2OCC2(C)C)=O)cnncc1O 95013,CC1(C)OC(=O)NC1C(N1CCN(C(=O)C(O)CC2CCCCC2)CC1)=O 95014,C1(C#N)(C(=O)NCC(CC)NC(=O)C(C)OCCN(C)C)CCC1 95015,Cc1ccc(C(N2CCC(C(C)NC(C3CC(=O)N(C4CC4)C3)=O)C2)=O)cn1 95016,CCCCC(C(=O)NCc1cc(=O)cc(C)[nH]1)NC(=O)C(SC)SC 95017,N1(C(c2c(CC)c[nH]c2)=O)CC(C)(C)CC1CNC(=O)Cc1n[nH]c(C)n1 95018,c1(C(N2CCCC(NC(=O)C3CC3)CC2)=O)cc2sccc2n1CC(F)(F)F 95019,c1(C(=O)OCC)cncc(C(=O)NCCCC(C)NC2CCN(CC(C)C)C2)c1 95020,c1(C(=O)NC(CNC(CNC(C(CC)C)=O)=O)(C)C2CC2)cc(S(N)(=O)=O)co1 95021,c1(SC)c(C(=O)NC(C)CNC(=O)COCc2nc(C)no2)cccc1F 95022,N1(C(C(CC)C)=O)CC(N)C(n2ccnn2)C1.c1(C(=O)C(=O)C2CC2)cc(C(N)=O)c[nH]1 95023,c1(CC(=O)NC(CN(C(=O)Cn2cc(CN(C)C)nn2)CC)C)ncccn1 95024,c1(CCC(=O)N(CC(C)NC(C(C2CC2)OCC)=O)C)ccncc1 95025,Cc1csc(=O)n1CC(=O)NCC1COC(CNC(C2CC(=CCO)C2)=O)C1 95026,Cc1cc(C(N2CCCC2CN(C)C(C2CC(F)C2)=O)=O)c2scnc2c1C 95027,c1(CN(C)C(C2CCCC2C(F)(F)F)=O)ccc(S(C)(=O)=O)cc1 95028,c1(C(N(CCC(=O)N(C(C#C)C)C)C)=O)cocc1C 95029,C1(CC(N2CCC(CC(C)NC(C3C(CCC)C3)=O)CC2)=O)CC2(CCC2)CO1 95030,N1(C(C(CC)OCC)=O)CCCN(C(=O)Cc2cccc(C(N)=O)c2)C(CO)C1 95031,C(CC(=O)N1CC(NC(C)=O)C1)(C(F)(F)F)NC(c1c(CC)ocn1)=O 95032,C1(NC(C2(CC=C)CCCC2)=O)CCN(C(=O)COCC(=C)C)CC1CO 95033,c1(C(=O)NCC2(NC(C3CCCCS3)=O)C(C)CCCC2)cc(O)c(O)c(O)c1 95034,C1(CNC(C2C(C)OC(=O)N2)=O)CN(C(C2(C)CCCCCC2)=O)CCCO1 95035,c1(C(N2CC(F)CC(NC(c3nc(OCC)oc3)=O)C2)=O)c[nH]nc1S(N)(=O)=O 95036,C1(C(=O)NC2C(NC(c3c(CC)scc3)=O)COCC2)CCCCC(=O)N1 95037,CC(C)(CCNC(C1(CC2CCC2)CC1)=O)NC(=O)CCCn1ccnn1 95038,N1(S(CCC)(=O)=O)CCC2(CCCC2C(=O)NCc2ccc3c(c2)OCO3)C1 95039,Cc1cc(O)c(Cl)cc1C(=O)N(C)CC1CCCN1C(c1cccc(F)c1F)=O 95040,CC1CC2CN(C(=O)CC(C)(C)N(C)C(C3COCC3(C)C)=O)CCN2C1 95041,N1(C(C2N(C(C(N3CCNC3=O)C)=O)C(C)CC2)=O)CCc2c[nH]nc2C1 95042,N1(C(C(=Cc2cnc[nH]2)C)=O)CCCC(NC(=O)Cn2cc(Br)c(C)n2)C1 95043,C1(N(C(C(F)=CCC)=O)CCNC(=O)C(c2ccccn2)C)CCCCCC1 95044,O=C(CCCNCCCCCNC(=O)NCCOC1C2COCC12)c1cccs1 95045,N1(C(C(F)OC)=O)CCC2(CC1)COCC(CNC(c1ncc[nH]c1=O)=O)O2 95046,N1(C(c2cc(-c3cccc(F)c3)on2)=O)CC2CC2(CNCc2ccsc2)C1 95047,C1(C(N(CC(=O)OC)C)=O)COCCN(C(=O)CC=C(Cl)Cl)C1 95048,C1(C(=O)NC2CC(c3c(F)cccc3F)C2)CN(C(=O)C(=O)C2CC2)CCC1O 95049,Cc1ccc(N2CCC2CNC(C2CCC(C3CC3)O2)=O)cc1.N1(C)C(=O)N1 95050,N1(C(C2OCCC(C)(C)C2)=O)CC(NC(c2cn[nH]c2)=O)C2(CCC2)C1 95051,C1(OC)COc2c(C(N3CCCC3CNC(c3nnsc3C)=O)=O)cnn2C1 95052,CC1CN(C(=O)NC(c2c(F)cccc2Cl)CO)CC1(F)F 95053,n1(CC)ncc(NC(C2CC(NC(c3cccnc3O)=O)C2(C)C)=O)c1C 95054,C1(CN(C)C(c2csc(-c3ccccn3)n2)=O)CCCN(C(=O)CCF)C1 95055,C(C(=O)NCC1(CNC(C2CCSC2)=O)CCC1)(C(C)C)OCC(C)C 95056,CN1CCCC(F)(C(=O)NC(C2CCCC2)CNC(c2cscc2Cl)=O)C1 95057,C(CCCCC(=O)NCCc1cnc(C)[nH]1)N(C(CNC(=O)OCC=C)=O)C 95058,C1(NC(CCNC(N)=O)=O)CCSC12CN(C(C1(NC(N)=O)CCOCC1)=O)C2 95059,C1(C(=O)NCC2(NC(C(c3c(C)cccc3)C)=O)CCC2)CC12CCOCC2 95060,N1(C(C2(CNC(c3nc(C)n(C)c3)=O)CC3(CC3)C2)=O)CCC2(CCOC2=O)C1 95061,S(=O)(=O)(c1ccc(NCC(C)O)c(F)c1)N(CC(C)N(C)C)C 95062,c1(C(=O)NC2CCCC(NC(c3n(C)cc(Cl)c3)=O)C2)cc(F)ccc1F 95063,N1(C(COc2ccc(SC)cc2)=O)CCCN(C(c2ccc(C(N)=O)[nH]2)=O)CC1 95064,c1(C(N2CC(C(C(=O)NC(C)CC3(O)CCC3)O)C2)=O)cnnn1C1CC1 95065,C(=O)(C(O)CC(C)(C)C)N1CCN(CCN(C(CC(C(=C)C)O)=O)C)CC1 95066,N1(C(=O)OC(C)(C)C)CC(O)CC1C(=O)NCCNC(c1conc1C1CC1)=O 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95084,C1(CNC(c2n(CC)ncn2)=O)(CC)CCCN1C(=O)CCC(=O)N(C)C 95085,CC1CN(C(C2(Cl)CC2(F)F)=O)CC(C(=O)NCCN=S(C)(C)=O)O1 95086,C=CC1(C(=O)NOCC(=O)NCC(=O)NCC(C)C)CCC1 95087,c1(C(=O)NCCNC(=O)CCC2CCCCCC2)cnn2c1OCC1(CC1)C2 95088,c12ccc(c(O)c1)c(=O)oc1nnc(s1)[nH]c(=O)[nH]2.CC(C)(C)OCCCCl 95089,CS(=O)(=O)CCC(=O)N1CC(CCCCNC(=O)Cc2ccccc2F)C1 95090,C(C(C)(C)CC(=O)NCCCOC1CCN(C(=O)C(O)C(C)C)CC1)OC 95091,c1(C(=O)NC(C)CC(=O)c2ccco2)cc(P(C)(C)=O)cs1 95092,c1(-c2cn(CC(C)NC(=O)CC34CCCC3C4)nn2)ccc2nc[nH]c2c1 95093,Cc1cc(F)c(C(=O)NCC2CCCN2C(c2cc3c(o2)CCCC3)=O)cc1F 95094,N1(C(C2CCN(C(C)=O)C2)=O)C2CCC1C(CO)N(C(c1ccc(C)s1)=O)C2 95095,Cc1[nH]c2ncccc2c1C(=O)NC12CC1CN(C(=O)COc1cnn(C)c1)C2 95096,C1(NC(C=C(C)Cl)=O)CC2CC(NC(c3nc(-c4cccs4)oc3C)=O)CC12 95097,CC1CN(C(c2nc(Cl)sc2Cl)C(=O)NC2COC2)CC1O 95098,C1(C)(C(=O)NCc2c(C(N(C)CC3C(C)OCC3)=O)[nH]cc2)CCN(C)C1 95099,C1(C)(NC(C2OCCC(NC(Cn3ncn(C)c3=O)=O)C2)=O)CCCCCC1 95100,Cc1ccc(NC(C2(F)CCN(c3cc(C)nc(C)n3)C2)=O)c(C#N)c1 95101,C12(C(=O)NCC(C)C)CC1CN(C(c1ccc(SC(F)(F)F)cc1)=O)C2 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95137,N1(C(CNC(CN(C(CC)=O)C2CCC2)=O)=O)CCC2(CCOCC2)C1 95138,C1(NC(C2(F)CN(C(Cn3ccc(C)c3)=O)C2)=O)CCC(CO)CC1 95139,n1(CC)cnc(C(=O)NCCN(CCOCCO)C(c2cc[nH]c2C)=O)c1 95140,N1(C(C2N(C)C(=O)CCC2)=O)CC2CCN(C(c3c(N)cnn3C)=O)CCC2C1 95141,c1(CC)c(C(N2CCC(CNC(c3cccc(CO)c3)=O)CC2)=O)cnn1CC 95142,CN(Cc1ccccc1N1CCCC1)N1CCC2(CNC(=O)N2)C1 95143,C1(C(C)C)CN(C(C2(O)CCCC2)=O)CCC1NC(c1n[nH]cc1C1CC1)=O 95144,c1(C(N(CC(=O)NCC(C)C)CC(C)C)=O)ccn2ccnc2c1 95145,C1(C(=O)NC(COC)(C)C)CC(F)(F)CN1c1nccc(C#N)n1 95146,c1(NC(c2c(NC(c3c(C)ccc(O)c3)=O)c[nH]n2)=O)ncnc2sccc12 95147,CCCCCC(O)CC(=O)NC1CN(C(c2ccc(OC(F)F)cc2)=O)CC1F 95148,c1(CSCC(=O)N(CC)CC)ccc2c(c1)OCCO2.C1(C)C(C)N1 95149,c1(C(C)NC(c2cccs2)=O)ccc(N(C2CCCC2)C(=O)CC2CCOC2)cc1 95150,C1(COC)(NC(c2nnn(C)c2C)=O)CCN(C(c2cnoc2C)=O)C1 95151,c1(C(=O)NCCCNC(CN2CCC(C)C2)=O)cnc([N+](=O)[O-])n1C 95152,C(=O)(CC1=CCOCC1)NCCn1cc(C(N2CCN(CCCC)CC2)=O)nn1 95153,C#CCCCC(C)C(=O)N1CCC(CCC(=O)NCC(C)(C)OC(C)C)C1 95154,N#Cc1cccc(CNC(N2CC3C(CC(=O)OC4C=CS(=O)(=O)C4)C3C2)=O)c1 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95226,CCC(F)(F)C(=O)NC(C1CC(NC(=O)CC2CCC(=O)NC2)C1)C 95227,N1(C(c2cc(OC)ncn2)=O)CCCC(CO)(NC(=O)CN(C)C(=O)C2CC2)C1 95228,c1(C(=O)NCCCCCC(=O)N(C2CCCC2C#N)C)cc2ccccc2[nH]1 95229,c1(C(N2C(C(=O)NC(CC)C(C)O)CC(F)C2)=O)ccc2cc[nH]c2c1Br 95230,n1(CCCN(CC(=O)N(C)CCOC2CC2)C)cc(-c2cnsc2)nn1 95231,C1(C(N2CCOCC2)=O)(N(C(C(F)=CCC)=O)C2CC2)CCSC1 95232,Cc1nn(C)c(Cl)c1CNC(c1ccccc1CN1CCCC(NC(N)=O)C1)=O 95233,N1(C(CC(C(=O)OC)(C)C)=O)CCCC2C1CCCN2C(c1ncncc1Cl)=O 95234,C12(C(=O)OC)C(NC(=O)NCCN3CCCC3C(N)=O)C3CC1C2C3 95235,N1(C(C2CCCC(C)C2)=O)CC(CNC(C2OCCCC2(C)C)=O)CC(C)C1 95236,C1(C(N(C(CCC)C(C)CC)CCC)=O)CCC2(CC2)CN1C(=O)OC(C)(C)C 95237,CC(C)S(=O)(=O)C(C)C(=O)NCC1(C(=O)Nc2cnccc2C(C)(C)C)CC1 95238,N1(C(C(COC)C)=O)C(C(=O)Nc2c(-c3ccccc3)nnn2C)CCC1C 95239,C1(NC(c2n[nH]c3c2COC3)=O)CN(C(c2cc(O)ncc2F)=O)C2CCCC12 95240,c1(C(C)S(N)(=O)=O)ccc(C(=O)OCCP(C)(C)=O)cc1 95241,N1(C(c2cccc(C)c2Cl)=O)CCN(C(=O)C(C)(O)CC(F)(F)F)CC12CCC2 95242,c1(C(N2CCC(C(C)NC(CCC)=O)CC2)=O)cc2cc(Cl)sc2[nH]1 95243,c1(CNC(=O)CCOCC(F)F)ncc(C(=O)NC(CO)C2CC2)cn1 95244,C1(NC(CCCOC)=O)CCCC(CNC(=O)CSc2cccc[n+]2[O-])C1 95245,c1(CS(CC(=O)N2CCOCC2)(=O)=O)cc2oc(-c3ccccc3)nc2cn1 95246,c1(CC)c(NC(=O)CC2CCN2C(C2(C)CCCCO2)=O)cnn1C 95247,C(=O)(C(C)C(C)(C)O)NCC(C1CC1)NC(c1nn(CC)c(C(F)(F)F)c1)=O 95248,N1(C(C(=O)NCC(C)O)=O)CCCC1c1ncc(-c2ccccc2)[nH]1 95249,Cc1cnn(CC(N2CCC3(CC3NC(=O)CC3COCC(C)O3)C2)=O)c(=O)c1 95250,c1(CC(=O)N(C2C(NC(CC=CC)=O)CCCC2)C)ccc(C)c(Cl)c1 95251,C1(CNC(C2CC23CCC3)=O)CCCN(C(c2cc(C3CCOCC3)no2)=O)C1 95252,c1(-c2nnc(C)o2)ccc(C(=O)NCC(CO)NC(=O)CCC=CC(C)C)cc1 95253,c1(NCCNC(C(=O)NC(c2ccoc2)C)=O)ccc(Cl)c(C(F)(F)F)c1 95254,O=C1NCCOc2c(Br)cc(C(N3CCC4(CC4)C3)=O)cc21 95255,c1(OC)cccc(Cl)c1CC(=O)N(C(C)CNC(=O)CC1COC(C)(C)CO1)C 95256,n1(CCCOC)nnnc1C(c1nncn1C(C)C)NC(COC)C(C)C 95257,C1(CC(=O)NCC(CCNC(C(CC)=CCCC)=O)O)CCCOCC1 95258,C1(NC(=O)C=Cc2cncs2)COC2(CCN(C(=O)Cc3cnns3)C2)C1 95259,Cc1cc(C(=O)NC(CNC(=O)C(C)Cc2ccc(F)cc2)C(C)C)nc(O)c1 95260,c1(NCc2ccc(C)nc2Cl)ccc(S(=O)(=O)NCC2COCO2)cc1Cl 95261,c1(C(=O)NC2C(NC(C(C3CCC3)OC)=O)C2)sccc1Cl 95262,C1(CNC(=O)Cc2csnc2Cl)CCN(C(C2(C(F)F)CC(O)C2)=O)CC1O 95263,Cc1coc(C(N2CCC(C3CCCN3C(=O)C(F)OC(F)(F)F)C2)=O)c1C 95264,n1(C(c2cccc(Br)c2)C#C)c(-c2cn(C)nn2)csc1=Nc1ccc(O)cc1 95265,C(c1cncnc1O)=CC(=O)NC(CCC)CNC(=O)CC1CN(C)C1 95266,C(CCCCCO)c1cn(CC(=O)NCCSCC2C(C)C2)nn1 95267,N1(C(c2cc(C)oc2)=O)CCCC(NC(=O)CC(C2CC2)C2CC2)C1C 95268,C1(CC(=O)N(C2CCCCC2)C)C2CN(C(=O)CC(F)F)CC12 95269,O=C(C1CCCn2nccc21)NC1(CO)CN(C(c2cc(F)c(F)cc2Cl)=O)C1 95270,c1(C(N(C)CC2CCN(C(CC3(OC)CCC3)=O)C2)=O)cc(C)ccc1C 95271,c1(NC2C(C(N)=O)CCC2)nc2ccccc2nc1NCCCO 95272,c1(C2(CN(C)CC3C(CC)CCC3)CCC2)ccc(Br)cc1 95273,c1(C(N(CCC(=O)N(CCCO)C)CC=C)=O)nn(C)cc1Cl 95274,C1(CNC(c2c(OC)csc2)=O)CN(C(=O)CCc2c[nH]c(=N)[nH]2)CC1C 95275,C(=O)(C1=C(F)CN(C(c2cccc(O)c2F)=O)CC1)NC1(C)CCCCC1 95276,N1(C(C(CCSC)NC(N)=O)=O)CCCC(CCNC(=O)C=C(C)C)CC1 95277,Cn1ncc(C(=O)NCC(CO)NC(=O)CC2CCN(CCF)CC2)c1Cl 95278,N1(C(COC(CC)C)=O)CC(C2CN(C(c3cc(C)c(OC)c(C)c3)=O)C2)C1 95279,N1(C(CCc2nc(C)c(C)o2)=O)CC(CO)C2(C1)CN(C(C1CC(F)(F)C1)=O)C2 95280,C1(OC)CN(C(=O)CC2OCCO2)CC1NC(=O)CC1(O)CC1 95281,c1(CC(=O)N(CCNC(=O)C(C)(CC)OC)CC)ccc([N+](=O)[O-])cc1Br 95282,Cc1ccc(CC(C)C(=O)NC(C)C(CO)NC(=O)CCC2CCCCC2)cc1 95283,C(=O)(C(=O)N1OC2CCC1C2)NCCc1ccc(OC)c(C(F)(F)F)c1 95284,c1(OC)ccc(CN2CC3CC3(C(=O)Nc3c[nH]nc3C)C2)nc1Br 95285,C1(C(=O)NCCCCCNC(c2[nH]n(C)c(=O)n2)=O)CCCC12NC(=O)NC2=O 95286,N1(C(C2CCC(COC)C2)=O)CC2(CCN(C(c3cc(C)sn3)=O)C2)C1 95287,C1(C(=O)NCCN2CCC(NC(C3C4CCCC34)=O)CC2)CCCCC1(F)F 95288,C1(CNC(C(C(C)C)F)=O)CC(C)CN(C(c2ccnn2C2CCCC2)=O)C1 95289,C1(C(N2CCC(C(C)NC(=O)Cn3cnnc3)CC2)=O)Cc2nccnc2C1 95290,N1(C(=O)COc2cccc(Br)c2)CCCC(C2CN(C(=O)C(F)F)C2)C1 95291,C(C)(CCC(=O)NC(C)(C)CN1CCN(C(=O)CCc2nnc(C)n2C)CC1)SC 95292,N1(C(C(C(C)OC)NC(c2c[nH]c(C#N)c2)=O)=O)CC2(C1)CC2(F)F 95293,C1(NC(CCSC)=O)CN(C(=O)COCC=Cc2ccccc2)CC12CC2 95294,Cc1ccc(F)c(C(N2CCC(O)(C(C)NC(=O)C=C3CCOCC3)C2)=O)c1Cl 95295,c1(CNC(C2(CNC(C3(C)CCCS3)=O)CCCC2)=O)cccc(CO)c1 95296,C(=O)(C1CCc2snnc21)NCCN(C(C)C)C(C1OCCOC1(C)C)=O 95297,C1(NC(C(C2CCCC2)NC(C(COC)C)=O)=O)CC2CCC1O2 95298,C=CCN=C(NCC=CC1CC1)NCC1C(C)(C)C1(F)F 95299,C1(NC(CN(CCC)C)=O)CCSC12CN(C(=O)C(C(C)C)n1cncn1)C2 95300,C(=O)(CC1=CCCCC1)NC1CN(C(C2CC3(CC(C)C3)C2)=O)CC12CC2 95301,C1(C(N2CCC3CC23C(=O)NCc2ccc(CO)o2)=O)CC2(CCCO2)C1 95302,c1(C(=O)NCC2CC(OC)CN2C(=O)CCCCC2CC2)c(C)nc(O)nc1C 95303,C=CCC(C)C(=O)NC1COCCC1C(=O)NCC(F)C1CCC1 95304,Cc1ccc(C2OCCCC2C(=O)NC2CC(=C3CC3)C2)cc1 95305,C1(C)(CN)CC(OC)CN1C(c1cnco1)=O.c1(C(=O)OCC)ccc(COC)cn1 95306,CC1(C)CCC(NC(=O)C=CC2CCCCC2)C(CNC(C2(C3CC3)CC2)=O)C1 95307,N1(C(c2ccc(NC)cc2)=O)CC2(C1)C(NC(=O)C(C)CC1CC1)CCS2(=O)=O 95308,Nc1ccc(Cl)cc1C(=O)NCC1(F)CC(NC(=O)CC2CCC(O)C2)C1 95309,C1(NC(CCCC(=O)NC(C)C)=O)COC2(CCN(C(C)C)C2)C1 95310,CC1(C)CCN(C(C2OCCC2(C)C)=O)CC1C(=O)NC1(CC(N)=O)CC1 95311,CN=C(NCCCn1cccn1)NC1CC(OC(C)(C)C)C1 95312,c1(CC(=O)NCC(C2CC2)NC(c2c(C(N)=O)coc2)=O)cnc2cccnn12 95313,C1(C(N(C2CN(C(=O)C(CO)N(C(=O)C(F)(F)F)C)C2)C)=O)CC2(C1)CC2F.CCO 95314,CC1(C)CCN(CCNC(C2C=CCCN2C(C2CCCC(=O)C2)=O)=O)C1 95315,Cc1c(CC(=O)NCC=C2CCN(C(=O)CCCCN(C)C)CC2)cnn1C 95316,CC1CCC(C(=O)NC2CC2CNC(c2ccnnc2O)=O)CC1 95317,c1(C(=O)NCCCOCCCNC(C2CCN(C)C2)=O)c[nH]c2ccncc12 95318,Cc1cc(N2CC(CC(C)NC(C3CCCCNC3=O)=O)C2)c(Br)cc1[N+](=O)[O-] 95319,Nc1cc(C(N2CCN(C(=O)C3=COCCC3)CC(O)C2)=O)c(F)c(F)c1F 95320,c1(C(N2CCCC(C)(NC(=O)CCC3(O)CCC3)C2)=O)ccc([N+](=O)[O-])cc1 95321,N1(C(c2c(SC)cc(F)cc2)=O)CC2CCN(C(c3cnc(N)c(N)c3)=O)C2C1 95322,c1(C(=O)NCc2nc(C(=O)NCCC3CC3)co2)cnc(O)c(F)c1 95323,C(=O)(C(F)C(CC)CC)N1C(CNC(CN(C2CC2)CC)=O)CCCCC1 95324,Cc1cnc(C(=O)NC2CCN(C(=O)C=CC3COC(C)(C)O3)C2)cc1Br 95325,c1(CCC(=O)NCC2N(C(c3occ(C)c3C)=O)CC2)c(Cl)cncc1Cl 95326,C1(NC(c2n(CC)ncn2)=O)C2CC3CN(C(=O)CNS(=O)(=O)CC)C1C3C2 95327,c1(C(=O)NCCC(C)NC(=O)CCOCC(F)(F)C(F)(F)F)cc(Cl)nnc1O 95328,c1(C(=O)NCCCOCCN(C)C(C2CC23CCOC3)=O)cn2cccnc2n1 95329,c1(C(N(C(C(=O)NC(C(=O)OCCC)(C)C)C)CCC)=O)ccc(CC)c(F)c1 95330,CCCC(C(O)C(=O)N1CCC(N(C)CC)C1)NC(=O)CCn1cnc(=N)[nH]1 95331,Cc1sc(N)c(C(N2CCC(NC(c3ccoc3Br)=O)C2)=O)c1C 95332,C(=O)(C1=CCCN(C(C2C=CC=CC=C2)=O)C1)N(CCCC)C 95333,CC1CCCc2c(C(=O)NC3(CNC(=O)CCN4CCCC4=O)CC3)cnn21 95334,CC1C(c2ccccc2)NCCN1C(C1CCC2CC2CC1)=O 95335,C12(C(N3C4C(NC(CC5(OCC)CC5)=O)CC(C4)C3)=O)CCC(CO)(CC1)CC2 95336,n1(CC)c(O)nc2cc(C(=O)NCC3CCC3NC(c3cnsn3)=O)ccc12 95337,C1(CC)COC(C)CN1C(c1nc(F)ccc1Br)C(=O)NC1CC(F)(F)C1 95338,C12(NC(C=CC(=O)N(C)C)=O)CCCCC1N(C(=O)Cc1csc(=N)[nH]1)CC2 95339,N1(CC(=O)NCC(CNC(CCOC(C)=O)=O)C)CCCCC1C 95340,CC1OCCCC1C(=O)NCCNC(=O)Cc1csc(-c2ccccn2)n1 95341,C1(CCC)CN(C(=O)CC2CCN(C(c3cc[nH]c(=N)n3)=O)C2)CCO1 95342,C(=O)(C(O)C(F)(F)F)N1CC(C(C)(C)O)(CNC(=O)Cc2ccccc2)C1 95343,c1(OC)ccc2c(ccn2CC(=O)NC2CCCC2CNC(=O)C(F)C(C)C)c1 95344,c1(C(=O)NCC2N(C(C3CCC3)=O)CCN(C)C2)nnc(O)c(Br)c1O 95345,C1(C(=O)NC2C(C)(C)C(Nc3ncc(Br)cn3)C2)CC2CCCCCCC12 95346,CC1CC(C(N2CC(NC(C3(C)CC3(F)Cl)=O)C2)=O)CCS1 95347,O=C1CC(c2ccc(C(=O)NCc3ccc(Cl)cn3)cc2)NC(=O)N1 95348,C(=O)(C(=O)N=S(C)(C)=O)N1CC(C)(c2cn(C3CC4OC(=O)CC34)nn2)C1 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95596,c1(N(C(C)CCNC(=O)CCCc2cccs2)C)ncnc(Cl)c1C#N 95597,c1(OC)ccc(CNC(=O)N(C)CCOc2c(C)cccc2C)cc1OC 95598,c1(CC)ccc(C(N2CC(C)CC2C(=O)NC2C3CCCOC23)=O)cc1 95599,Cc1cccc(C(=O)NC2(C)CC(NC(=O)C(C3CC(F)(F)C3)O)C2)c1 95600,C1(C(N(C(C)CS(C)(=O)=O)C)=O)CN(C(=O)OC(C)(C)C)CC12C(=O)NCC2 95601,N1(C(=O)NCC2CC3(CC(OC4(C)CCCCC4)C3)C2)CC2OCCOC2C1 95602,c1(C(=O)NCC(CN(C(C2(CSC)CC2)=O)C)O)cn(C)cc1C(F)(F)F 95603,c1(C(=O)NCC(=CC(=O)NC(C(COC)C)C)C)c(C)cccc1F 95604,N(C1CCC(NC(c2sccc2C#N)=O)c2ccccc21)C(C=C(CC)C)=O 95605,c1(NCCCCNC(c2cnn(C3CCCC3)c2)=O)ncnc(Cl)c1CO 95606,N1(CC(=O)NCC2CN(C(C(OC)OC)=O)C(C)CC2)C(=O)CC(C)(C)C1=O 95607,c1(CC)cc(C(=O)NC(c2ncc(C(=O)OC)s2)C)sc1CC 95608,N1(C(CNC(=O)OCC)=O)CCOCC(C)(CNC(=O)C(C)C2CCCO2)C1 95609,C1(CC(N2CCCC(CNC(c3nncs3)=O)C2)=O)CC(c2ccccc2)=NO1 95610,C=CCC(C)(C)C(=O)NCCC1(OC)CCC1.c12cnc(s1)CNC2=O 95611,CCC(C(=O)NCC(C)NC(c1ccc2nccn2c1)=O)C(C)(F)F 95612,c1(CC(=O)NC2C(NC(C(C)OC(C)(C)C)=O)C(O)C2)cncnc1O 95613,c1(C(=O)NCCCC(=O)NC2(CC=C)CC2)cncc(OCC)c1 95614,C1(C(=O)Nc2cccc(C3(C)CC3)c2)CC2CCCCN2C1=O 95615,C(C1=CCN(C(=O)C=Cc2cncc(OC)c2)CC1)NC(C1N(CC)CCC1)=O 95616,c1(OC)ccccc1-c1ccnc(NC2CCN(C(C3CCOC3C)=O)C2)n1 95617,C(=O)(C(F)(F)c1ccccn1)NCC(C)(C1CC1)NC(=O)C(O)CN1CCCC1 95618,CCCC(C)CC(=O)N1CC(NC(c2ccnc(Cl)c2O)=O)C(C)C1 95619,Nc1ccccc1-c1cn(CCCC(=O)NCCc2csc(O)n2)nn1 95620,c1(-c2ccc(C(CC)=O)s2)cccc(CNCc2cnc(C(=O)O)o2)c1 95621,C(CCSC)(C(=O)N1CCC1C(=O)NOCc1cnn(C(F)F)c1)OC 95622,c1(C(=O)NCC(C)NC(=O)C(C2CC2)N(C)C)cc(-c2cccnc2)on1 95623,O=S(=O)(c1ccc(N2CCC3(CCC3)C2)cc1Br)NCC1C2CCCCC12 95624,N1(C(c2ncc(F)cc2I)=O)CCc2c(O)ncnc2C1 95625,c1(C(C(=O)Nc2ccccc2Cl)N(CCOCC)CC)ccc(F)c(OC)c1 95626,C1(C(=O)Nc2cc(C)c(-c3ccncc3)cc2)C2Cc3ccc(Cl)cc3C12 95627,C1(CC(=O)NCCN(C)C(C2CC2C(N)=O)=O)CCCCO1 95628,C1(C(N2C(CC(=O)N(C)Cc3cccc(O)c3)COCC2)=O)OCCN(C)C1=O 95629,N1(CC(CNc2ccc(CN(C3CCOCC3)CC)cc2)O)CCC(F)(F)C(C)C1 95630,CC1CN(C(c2ccc(NCc3ccc(Br)o3)cn2)=O)CCN1C 95631,CCC(CC(=O)N1CCC(C2CC2)(CNC(c2cnsc2)=O)C1)C(F)F 95632,Cc1ncc2n1CCC(C(N1CC(C)(C)OCC1CNC(=O)C(C)(C)C#N)=O)C2 95633,C1(C(N2CC(C(=O)NC(C=C)(C)CC)C(OC)C2)=O)OCCCC1(C)C 95634,N1(C(c2cnc(CNC(C(CCCC)N(C)C)=O)nc2)=O)CCN(C)C(=O)C1C 95635,c1(C(N2CCCC(C(C)NC(CCC(=O)OCC)=O)C2)=O)nnn2c1CCCC2 95636,C(=O)(C(O)CCNC(c1ccc(N)cn1)=O)NC(COC(C)=O)CO 95637,Cc1cc(C)c(C(N2CCC(C)(NC(=O)CC3NC(=O)NC3=O)C2)=O)[nH]1 95638,Cc1nc(N2CC3CC2CN(C(=O)CCC(C)N(C)C)C3)ccc1[N+](=O)[O-] 95639,CC(CCN=c1nc(-n2ccnc2)cc[nH]1)NC(=O)CC1CCN(C)C1=O 95640,N1(C(c2ccc(C)c(Cl)c2)=O)CCCC2C1CCN2C(C1CC2C=CC1O2)=O 95641,Cc1cn2ccc(C(=O)NCC(C)(C(C)C)NC(c3cnnc(O)c3)=O)cc2n1 95642,C1(C(N2CC(CCNC(c3n[nH]cc3C3CCC3)=O)C2)=O)CCc2nncn2C1 95643,N1(C(C(C)OC)=O)CC2C(C(=O)NC3CC(C(C)(C)C)C3)C2C1 95644,N1(C(c2ccc(C(F)F)cc2Cl)C(=O)NC)CC2(CCC2)CCC1C 95645,c1(C(N2C(CCNC(CC(C)OC)=O)CSCC2)=O)c(F)cc(OC)cc1F 95646,c1(C(=O)NC2CCN(C(C(COCC)(C)C)=O)CC2)ncc(OC)cc1F 95647,c1(C(N(CC(C)O)CCNC(C23CC(F)(C2)C3)=O)=O)cccc(OC(C)(C)C)n1 95648,C12(C(=O)N(Cc3cc(C4CCCC4)no3)CC)CC1CCN2Cc1ccc(Br)o1 95649,C1(C(=O)NCCN(C(C=CC=CC)=O)CCOCCO)CCCC2(CCC2)O1 95650,c1(OCCCC)ccc(CNCc2ccn(CC(F)(F)F)n2)cc1OC 95651,c1(OC)ccc(-n2nc(C(C)C)nc2CCCCCN(C)C)cc1F 95652,c1(C(=O)NCC(CNC(C(C=CC)O)=O)C(F)(F)F)cncc(P(C)(C)=O)c1 95653,c1(-c2n(C34CC(C)(OC3)C4)ccn2)ccc2c(c1)CCO2 95654,N1(C(=O)CNCc2nccs2)CC(OC)C(OC)C1CNC(C1(C2CC2)CC1)=O 95655,C#CCCCCCCC(=O)NCCCNC(=O)CCn1cc([N+](=O)[O-])cn1 95656,Cc1nn(C)c(Cl)c1C(N1CCN(C(C2(COC(C)C)CC2)=O)CC1C)=O 95657,Cc1nn(C)c(C)c1CC(=O)NCC1CC(F)(CNC(=O)CC2(C)CC2(F)Cl)C1 95658,Cc1nn(C)c(C)c1OCC(=O)NCCC1CCC(NC(c2scnc2C)=O)C1 95659,C(=O)(C(F)(F)C(F)(F)F)NCCNC(c1cc[nH]c1)=O 95660,C(=O)(CC(C(C)(C)C)NC(=O)C(C)CC#N)NCC1CCN(C(C)C)C1 95661,N1(C(C(CC=C)C)=O)CC(C(=O)NC2CCC3(CC2)N=N3)CCC1(C)C 95662,C(=O)(CC(C)(C)N1CCC1)NC(C(C)OC1(C(=O)Nc2ccccc2)CC1)C 95663,C1(CCC(=O)NCCC(=C)CNC(=O)CN2CCCCC2)C(=O)NN=C1C 95664,CCC(C)C(CNC(C1CSCN1C(C1(CC)CCC1)=O)=O)CO 95665,C1(NC(C(CC)Oc2ccccc2)=O)CCCC(CNC(=O)C(F)=CCCF)C1 95666,c1(C(=O)NC(C(C)NC(=O)C(C2(O)CCCC2)F)C)cnn2ccn(C)c12 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95859,CC1C=C(C(=O)NC2CCCC(NC(C3C4CCCCC34)=O)C2)C1 95860,N(C(=NCCCCl)NC1CCCCC1)Cc1nnn(C)n1 95861,C1(C)(C(=O)NC2CC(NC(c3ccc(CNC(C)=O)s3)=O)C2)COCCO1 95862,N=C1NC(=O)C(CC(N2CC(CNC(=O)CC3(O)CCC3)C2)=O)S1 95863,C=CCC(C)(C)CC(=O)NCC(C)(O)CNC(C1CC(=O)CCO1)=O 95864,C(=O)(C1c2c[nH]nc2CN1C(c1snc(C)c1N)=O)N(CC#C)CC1CC1 95865,CC1CC(NC(c2ccc(C#N)o2)=O)CCN1C(=O)CCc1cnccn1 95866,C1(CC=C)(C(=O)NCCCOc2cccc(O)c2)CCCN1C(=O)CC1(C)CC1 95867,c1(C(=O)NC23CC(CNC(C4C(C)(CC)C4)=O)(OC2)C3)cc(OC)c(F)c(F)c1 95868,C#CCC(C)(C(=O)N(CCSC)CC)NC(c1ccc(C)c(C)c1)=O 95869,C1(C)(C(=O)NCCC2(O)CN(C(C(C)c3cccs3)=O)C2)CCC(=O)N(C)C1 95870,Cc1cccc(C(N2CC(C(C)NC(c3cccc(Cl)c3)=O)C2)=O)c1N 95871,N1(C(C(Cn2ccc(C)cc2=O)(C)O)=O)CCCC2COCCC12 95872,C1(C(=O)NCC(C2CC2)NC(CC=C=C)=O)COC=CN1C(=O)OC(C)(C)C 95873,N1(C(C(C2CCOCC2)OCC)=O)CCCC(NC(=O)C(C)OCCOC)CC1 95874,c1(C(=O)NCCC2CCN(C(=O)Cc3ccoc3)C2)cnc(-n2cccn2)cn1 95875,C1(CNC(C(C(C)C)C)=O)C2CCC(C2)N1C(=O)CN(C)Cc1ccccc1 95876,C=C(Cl)C(C)(C)C(=O)NCC1(F)CC(CNC(C2OCC2(C)C)=O)C1 95877,c1(C(CNC(C2CC(OC)C2)=O)NC(=O)CCOC)ccc(F)cc1 95878,C#CCC(C)(C)C(=O)NCC1(O)CC(CNC(=O)C=Cc2ccc(O)cc2)C1 95879,Fc1cc(NC(c2cccc(I)c2)c2nnnn2C2CC2)cc(Br)c1 95880,C1(COC)CN(C(C2(NC(c3coc(C)n3)=O)CC2(C)C)=O)CCO1 95881,Cc1nn(C(C)(C)C)cc1C(=O)NC1CCC(C)(CNC(=O)CC(F)(F)F)C1 95882,Cc1cc(=NC(=O)CNC(CSCC23CCCN(C(=O)CC4CC4)C2C3)=O)[nH]o1 95883,c1(C(N2C3(CNC(=O)COCC4CCCO4)CC(C2)C3)=O)cccc(Cl)c1Cl 95884,C(=O)(C1=CC2C=CC1C2)NC1C2CC(C(=O)NCCC(C(=O)OC)C)C(C2)C1 95885,c1(C(N2CCC(N(C(=O)CN3CCNC3=O)CCC)C2)=O)oc(COC)nc1C 95886,c1(C(N2CC3C(N(C(C4C(OC)CCC4)=O)C)C3C2)=O)sc2ncccc2c1N 95887,CC1(C(=O)NCC#CCNC(=O)Cc2cccc(C(N)=O)c2)CC2CCC1C2 95888,C1(NC(c2c(OC)cccc2)=O)CN(C(C2(CCO)CC2)=O)CCC1C 95889,C(C)(C)(CC(F)C(=O)NCCNC(=O)N(C)C)NC(C1ON=C(C(C)C)C1)=O 95890,n1(CC(=O)NCCC(C)NC(CC2CC(=C)C2)=O)c(=O)nc(O)c2ccccc12 95891,C1(CNC(C2(C)CCN(C(COCCCC(C)C)=O)C2)=O)CCC2(CCC2)O1 95892,Cc1ccnc(O)c1C(=O)NC1CCCCCC1NC(=O)Cc1sc(O)nc1O 95893,C1(NC(c2sccc2Br)=O)CN(C(c2c[nH]nc2F)=O)CC1O 95894,C1(NC(C2ON=C(CC)C2)=O)CCCCCC1C(N1CC(C(=O)NC)(OC)C1)=O 95895,C(=O)(C(C(C)(C)C)C1CCCC1)NCCN(C(C1CCN(C)C1=O)=O)C 95896,c1(CNC(C(C(C)C)OC)=O)cccc2c1CCN(C(=O)CC1(OC)CCC1)C2 95897,CC1(C)CC(C)(C(N2CC(F)(C3CC3)C2)=O)CN1C(=O)Cc1ccon1 95898,CC(CC(=O)NC(CNC(=O)CN1CC2CC2C1)CO)NC(C1CCCC1)=O 95899,C1(C(C)NC(=O)C(C)(C)c2ncco2)CCCN(C(=O)CCCCNC(N)=O)C1 95900,C(=O)(CCCC(F)(F)Br)N(C1CCN(C(C2CC(C)(C)CO2)=O)C1)C 95901,N1(C(C(CSC)OC)=O)CC2CCC1C(CNC(=O)C=CC(C)(C)C)C2 95902,N1(C(COC(C)=O)=O)CCN(C)C(C(=O)NC(c2cccnc2C)C)C1 95903,C1(C(=O)NCC2CC(NC(C3(C#N)CC(C)C3)=O)C2)CCOC(C)(C)C1 95904,N1(C(C(C)=C2CCC2)=O)CCN(C(=O)CCc2n[nH]c3ccccc23)CC(O)C1 95905,CCCCCCC(O)CCC(=O)NC1CCN(C(=O)C=CS(=O)(=O)CC)CC1C 95906,CC1CC(C(=O)NC2CN(C)CC2O)N(C(=O)OCc2ccccc2)C1 95907,C(Cn1cc(CN(C)CCOC)nn1)(CC(C)C)NC(C1C(C=C)C1)=O 95908,N1(C(C2CC(=C)C2)=O)CC(NC(=O)CCOCC(F)(F)C(F)(F)F)CC(O)C1 95909,CC1CN2CCN1C(C(N1CCC(N(C)C(c3nccn4nccc34)=O)C1)=O)C2 95910,N1(C(=O)Nc2ncnc(O)c2Br)CCC2(C(=O)O)C(C1)C2(F)F 95911,c1(C(C(=O)NC2(C)CC2)N(CCC#C)C2CC2)ccc([N+](=O)[O-])c(O)c1 95912,N1(C(c2c(O)ccc(SC)c2)=O)CC2CCC(NC(c3ccsc3)=O)CC2C1 95913,C=C(C)c1cccc(NC(C2C(C)OCCN2C(=O)CC(C)(C)C#N)=O)c1 95914,C(C(C)(O)C(F)(F)F)NC(=O)Nc1ccc(NC(=O)OC(C)(C)C)nc1 95915,C1(NC(C(C)N(c2ccccc2)CC=C)=O)COCCN(C(=O)C=CC=C(Cl)Cl)C1 95916,CC1(C)OCCCC1NC(=O)CC1CCN(C(=O)CNc2ccccn2)CC1 95917,N1(C(C)=O)CCC(N(C(=O)CC2(CNC(=O)C(C)n3cncn3)CC2)C)C1 95918,c1(CCCC(=O)NCC(CNC(CN(C2CCC2)C)=O)F)csc2ccccc12 95919,C1(C(C(=O)NC(CCC)CO)C)CCCN(C(=O)CCCn2cccn2)C1 95920,CC1CN(C(=O)CN(C)C(N)=O)CC(CCNC(=O)C(c2ccccc2F)O)O1 95921,c1(C(N2CC(N3CCN(C(C(CCSC)O)=O)CC3)C2)=O)cc2n(n1)CCO2 95922,c1(CCCC(=O)NC2C=CCN(C(CSCC(=O)OC)=O)C2)ccc(C)c(C)c1 95923,Cn1cc(C(=O)NCC2(C)CCCN2c2cc(C3CC3)nc(Cl)n2)n(C)c1=O 95924,N1(C(C2(F)C(C)OCC2)=O)CCCC2(CCN(C(=O)CC3CCC=CCC3)C2)C1 95925,c1(C(=O)NCCCCNC(C2COC(=O)O2)=O)ccc2cncnc2c1 95926,c1(C(=O)NCC(C)NC(=O)C2=CCSC2)c[nH]c2cccc(C#N)c12 95927,N1(C(c2cc(C(F)(F)F)ccc2I)=O)CCC2(CCN(Cc3cccnn3)C2)C1 95928,N1(C(c2ccc(C(=O)OCC)cc2)=O)CCN(C(=O)C(C)C(C)(C)C)CC(O)C1 95929,C1(C(=O)NCC(c2ccc(F)cc2)NC(=O)C(F)C2CCC2)CCCCS1(=O)=O 95930,c1(C(C)(C)CNC(=O)OCc2nc[nH]n2)ccc(F)cn1 95931,C(=O)(C(CC(F)F)C1CCC1)NCCN(C(C1(C)ON=C(C)C1)=O)C 95932,CC(C)(C(=O)NCC(CO)NC(C1CCOC1)=O)C1CCC1 95933,C1(NC(C2(C(=O)OC)CC23CCC3)=O)C2CC3CC1CC(O)(C3)C2 95934,CNS(=O)(=O)N1CCC(C(=O)NCCNC(C2CN3CCCN2CC3)=O)CC1 95935,C1(c2ccccc2)(NC(C(C)=CC)=O)CCN(C(=O)C=Cc2nccs2)C1 95936,CC1CCC(Cl)=C(C(=O)N2CCN(C(=O)C(C)(C)CS(N)(=O)=O)CC(C)(C)C2)C1 95937,N1(C(c2c(C)csc2)=O)CC2CC(C1)CN(C(C1CC(C)(C)C(C)(C)C1)=O)C2 95938,c1(C(N2CCOCC(NC(C(COC)(F)F)=O)C2)=O)cc2ccc(F)cc2cn1 95939,c1(C(N2C(CNC(c3ccc(OC)nc3)=O)CC2)=O)ccc(F)c2ccsc12 95940,C1(N(C(c2cc(C(C)C)no2)=O)C)CCCC(NC(C2(CCN(C)C)CC2)=O)C1 95941,c1(CC(=O)NCC(CC)(C)NC(C2CNC(=O)C2)=O)nc2ncccn2n1 95942,Cc1cccc(F)c1CNC(=O)C(C)N(C(=O)CC1CCCC(C)O1)C 95943,N=c1cc[nH]cc1CNC(C1CCN(c2ccc(-c3cn[nH]c3)cc2)CC1)=O 95944,C1(CNC(Cc2cccc(OCC)c2)=O)CN(C(c2scnc2C)=O)CC12CC2 95945,CN(CCCC(=O)NCC1C2CN(C(=O)C(O)C(F)(F)F)CC12)N=O 95946,c1(SC)cccc(C(=O)NC2CN(C(c3cccnc3O)=O)CC2C)c1O 95947,O=C1CCC(C(=O)N2CC3(NC(=O)CC4CCCC(=O)N4)CC2C3)=NN1 95948,Cc1onc(C(N2CCCC(NC(c3cc(Br)no3)=O)C2)=O)c1[N+](=O)[O-] 95949,c1(C(C)OC(c2ccc(OC)o2)=O)ccnc(SCC(=O)NN2CCOCC2)c1 95950,c1(N2CC(C)(C)OCC2)nc2cccnc2c(=NC2CCC(CCCCCl)C2)[nH]1 95951,N1(C(C(C)CC(C)(C)C)=O)CC(CNC(c2cccn2C)=O)C2(CCOCC2)C1 95952,C1(NC(c2ccnc(NC3CC3)c2)=O)(CNC(C2(CCO)CC2)=O)CCCCC1 95953,C12(C(N(C)Cc3ccnn3C)=O)CCCC1CN(C(C1(C#N)CCCCC1)=O)C2 95954,c1(CC(=O)NCC2CN(C(=O)C(O)C3CCC3)C2)cccc(-c2nnco2)c1 95955,N1(C(C(CC(C)C)ONC(C2CCOCC2(C)C)=O)=O)CCc2c(nnn2C)C1 95956,c1(C(=O)Oc2cccc(CN=c3nnn(C)[nH]3)c2)oc2ccccc2c1CO 95957,C1(C(N2CC3C(NC(C(C)N(C(C)=O)C)=O)C3C2)=O)CCC([N+](=O)[O-])CC1 95958,c1(CC(C)NC(c2cc(Cl)ns2)=O)ccc(CNC(=O)CC2(C)CC2)cc1 95959,C(CC(=O)N1CC2CCC(C1)N2C(=O)C=Cc1ncc[nH]1)(C(F)(F)F)OC 95960,C1(C(=O)NC(C(=O)NC)CC2CC2)CCC(C2CC2)N1C(C1CC(F)CN1C)=O 95961,N1(C(c2cnc(COC)s2)=O)CC2(CCC2NC(=O)C=C(C)Cl)C1 95962,c1(CCC(=O)NCC(C)(C)NC(C=CCCC)=O)ccc(O)c(Cl)c1 95963,N1(C(C2(C)COC2)=O)CCCC2(CCCCC2NC(C2CC3CC3C2)=O)C1 95964,Cc1cc(C(N2CCC(C(C)C(=O)N(C3CCCCC3O)C)CC2)=O)cc(C)n1 95965,N1(C(C2CCC(C)C2)=O)CC2C(CNC(c3cc(O)nn3C)=O)C2C1 95966,N1(C(CCC(C)(C)NC(CCCOCCOC)=O)=O)CC2CCCCCC2C1 95967,CN1C(=O)Cc2c(C(=O)NC(Cc3ccc(Br)c(C)c3)C(=O)O)cccc21 95968,C(=O)(CC(C)(C)C)N(CCC=C)CC1CCC(Oc2ccncc2)C1 95969,CC(C)(C)CC(O)C(=O)N1CCCC1CNC(c1ncc2[nH]ncc2n1)=O 95970,N1(C(C2(C3CCCO3)CC2)=O)CCCCC1C(=O)N(C)CC1(CC)CC1 95971,C(CC(C(=O)N1CCOC(CCCNC(=O)C(Br)=C(C)C)C1)OC)OC 95972,c1(C(N(C(C)C(N2CCCC(C)(C)C2C)=O)CC)=O)ccc2[nH]ccc2c1 95973,CCC(CC(F)(F)F)C(=O)N(CCC(C)NC(c1cnc(Cl)s1)=O)C 95974,c1(C(N2C3(CNC(CC4(C)CC4(Cl)Cl)=O)CC(C2)C3)=O)cccc2c[nH]nc12 95975,N1(C(c2c(COC)ccs2)=O)CCN(C(=O)C=Cc2cscn2)C(CC(F)F)C1 95976,c1(NC(N2C(CNC(c3cc(COC)on3)=O)CC2)=O)cc(C)ccc1[N+](=O)[O-] 95977,Cc1nc(NC2CC2)sc1C(=O)NC(C)CN(C)C(C1CC2CC2C1)=O 95978,C(CC(C)(C)C)(C(=O)NC1CCCCC1C(=O)N(C)Cc1cnccn1)OC 95979,c1(-c2ccc(C)cc2)ccc2c(c1)C(C(=O)O)OCC2 95980,c1(CC)cc(C(N2CCCC2C(C)NC(c2cc(F)ccc2F)=O)=O)ccc1Cl 95981,c1(C(=O)NC2C(C)CN(C(=O)CCCN(C)N=O)C2)noc2c1CC(C)(C)CC2 95982,C#CCC(C)(C)C(=O)NC1CC(N(C(=O)CCC=CC(C)C)C)C1 95983,c1(OC)cnnc(C(=O)NC2CC3(C2)CC3C(=O)NC2CN(c3ncco3)C2)c1 95984,O=C(CN1C(=O)C(F)(F)Oc2ccccc21)OC(C(F)(F)F)c1nccs1 95985,C1(CNC(C2CCC(C)CC2)=O)CCN(C(=O)Cc2cc(Cl)ccc2O)C1(C)C 95986,CC(CC(N)=O)C(=O)N1CCCC(C(CC2CC2)N=c2[nH]ncs2)C1 95987,C1(C(=O)NC2CC(F)(CO)C2)C2CN(C(=O)CSCc3ccc(F)cc3)CC12 95988,C(=O)(NNc1cc(Cl)cc(Cl)c1)NC1COCCN(Cc2c(C)ccc(C)c2)C1 95989,n1(CCCN(C)C)nc(-c2ccc(N)cn2)nc1CCN1CCCC1=O 95990,C1(C2C(OCCC(=O)NC3CC3)C2)CCCN(C(c2cncc(C3CC3)c2)=O)C1 95991,N1(C(C(C)=O)=O)CCCC(C)C1CNC(=O)CCc1cn(C)nn1 95992,C1(NC(CC(C)F)=O)CN(C(=O)CCOc2cccnc2)C2(CCCC2)C1 95993,C(CCC(O)CO)NC(C1CC(CNC(C2(CO)CCCO2)=O)OC1)=O 95994,C1(NC(c2cc(OC)c(Cl)cc2)=O)CCC2CN(C(c3nncn3C)C)CC2C1 95995,c1(C(=O)NC2CCC(C)(CNC(c3c(C)nn(C)c3)=O)C2)cccc([N+](=O)[O-])c1 95996,c1(SC)ccc(Cl)c(C(N2CCN(CCc3cn(C(C)C)nn3)CC2)=O)c1 95997,CC(C)C(C)CC(=O)N1CC(O)CC1CNC(=O)COc1ccon1 95998,N1(C(CC2CCCC(C)(C)O2)=O)CCN(C(=O)CC(F)(F)F)CC12CCC2 95999,N1(CC(=O)Nc2cccc(C(C)C)c2)CC2CN(S(=O)(=O)C(F)(F)F)CC12 96000,C1(NC(C2CC(CC)(CC)C2)=O)C=CCN(C(=O)C(N2CCOCC2)C)C1 96001,c1(NC(C2C(C(=O)Nc3c(OC)cccc3)C2)=O)ccc(S(C)(=O)=O)c(F)c1 96002,Cc1c(C(N2CC3CC3(CNC(C3(C)CC4CC4C3)=O)C2)=O)cccc1C1CC1 96003,N1(C(C(C)(C)OCC)=O)CCCC(C(=O)NCc2nc(CO)n[nH]2)C1 96004,C(C)(CNC(c1ccc(-c2cccs2)o1)=O)(CO)NC(C=C(CCC)C)=O 96005,c1(OC)ccc(C(N2CCC(CNC(c3cccc(Cl)c3I)=O)C2)=O)c(Br)n1 96006,c1(C(=O)NCC2C(CNC(C(F)=CC)=O)C2)ccc(-c2cccnc2)s1 96007,c1(C(=O)NCCn2cc(C(=O)NC(COC)C3CCC3)nn2)cncc(C)n1 96008,c1(NC(C(C)n2ccnn2)=O)cccc(CNC(c2ccoc2Br)=O)c1 96009,c1(OC)c(F)c(CNc2ncnc(NC(C)CF)c2C)cc(F)c1F 96010,C1(C(=O)NCc2c(C(=O)NC3CCN(C)C3)occ2)CC1C1CCCC1 96011,N1(C(c2c(C)ccs2)=O)CCN(C(C2CCN(CC(F)(F)F)C2)=O)CC2(CC2)C1 96012,C1(C(=O)NCCC2(C(=O)NC3(CN(C)C)CCC3)CC2)CCC(C)(C)C1 96013,C(=O)(CC(C)(C)CC(F)F)NC1CC(C)N(C(C2CCN2C2CCCC2)=O)C1 96014,Cc1cccc(C(=O)NCC2(C)CCC(NC(c3cnccn3)=O)C2)c1 96015,C1(C#N)(C(=O)NCC2CC(OC)CN2C(C2CCC2(C)C)=O)CCOCC1 96016,C1(C(=O)NCCSCCC=C)CCC(O)CN1C(c1cccc(OC)n1)=O 96017,C12(NC(CN(CCC)C)=O)CC(CNC(=O)CCC(C)(C)OC)(C1)OC21CCC1 96018,c1(C(N(C(CCC)C)C)=O)ccn(CCNC(=O)CC2(C)CCCO2)c1 96019,N#Cc1cc(Br)ccc1CN1CC2CN(c3ncc(C4CC4)cn3)CC2C1 96020,N1(C(C2(C)C(C)C2)=O)CCOCC(CNC(c2ccc(Cl)c(Cl)c2)=O)C1 96021,n1(CC(N2CCCC2c2cc(C3CC3)on2)=O)ccc(C(F)F)n1 96022,N1(CC(=O)N(CC(CC)NC(=O)C(F)=CC2CC2)C)C(=O)NC2(CCCC2)C1=O 96023,N1(C(=O)NCc2ccc(C)cc2OCC(F)F)CC2C3C=CC(C3)C2C1 96024,C(C(=O)N=c1ccn(C(C)C)[nH]1)(c1cccs1)NC(c1c(C)cns1)=O 96025,c1(-c2cccc(CO)c2F)ccc2nccn2n1 96026,CN=c1[nH]c(=NCCCN2CCN(C)CC2)[nH]c(=NC2CCSCC2)[nH]1 96027,C#CC(C(C)(C)C)NC(=O)COCCNC(c1cccc(CC)n1)=O 96028,C(=O)(C(C)Cc1cnc[nH]1)NCCN(CCOC)C(C1(n2cncn2)CC1)=O 96029,C(CC1C(=O)Nc2ccccc21)NC(=NCCCC)NC(C)CCC(F)F 96030,C1(NC(C2(NC(C)C)CC2)=O)COC2(C1)CN(C(=O)C(N1CCCCC1)C)C2 96031,C1(CCC)CN(C(C2CCCCN2CCC)=O)CCN1C(=O)C1=CCC1 96032,C(=O)(C(C(=O)NCCn1ccc(C(=O)NC23CC(C)(C2)C3)c1)OC)OCC 96033,c1(N2C3C(CNC(C4(C)CC4Br)=O)C(CCC3)C2)nc(O)c2ccc(Cl)cc2n1 96034,c1(NC)cncc(C(=O)NC2CCC(N(C)C(c3ccc(C(N)=O)[nH]3)=O)CC2)c1 96035,c1(C(C(C)NC(=O)CCc2cnc[nH]2)NC(=O)CSc2nncs2)ccccc1 96036,C1(CNC(CCC(CC)C)=O)CC2(CO1)CN(C(=O)CC1CCCCC1)C2 96037,N1(C(C(COC)Cl)=O)CC(NC(c2cc(Br)c[nH]2)=O)C2(COC2)C1 96038,C=CCN(OC)C(=O)C(C)N(C(=O)CCCN1CCCC1)C 96039,c1(C(N2CCCC2C(C)(C)N)C(=O)NC(CC)(C)C)cnc(OC)c(F)c1 96040,C(=O)(C#Cc1ccccc1)NC1CCCN(Cc2c(C)c[nH]n2)CC1 96041,C1(C(N(CCCCC(=O)NC(CC(=C)C)CO)C)=O)CC2CC1CC2=O 96042,CCN=c1[nH]c(C(=O)NCCC(C)(C)CNC(c2cnc(O)cc2OC)=O)cs1 96043,C#CCCCCC(=O)NCC12CC(NC(C3CCCC3(F)F)=O)(C1)C2 96044,C1(C2CCOC2)(C(N(CCN(C(C(C2CC2)OC)=O)C)C)=O)CCOCC1 96045,c1(C(=O)NCC(=O)N(CCCN(CC)CC)C)cc(O)cc(=O)o1 96046,C(=O)(CCNC(=O)C(C1CCOC1)NC(=O)CCn1cnnn1)OC 96047,c1(C2(C(=O)NC(C3CN(C(C4(F)CCOC4C)=O)CCO3)C)CC2)ccc(F)cc1 96048,CC1CCN(C(C2(C(F)(F)F)CC(O)C2)=O)CCN1C(c1scnc1Cl)=O 96049,N1(C(c2c(CC(=O)OC)occ2)=O)CC(NC(c2cc(C)c(C)[nH]2)=O)CC2(CC2)C1 96050,c1(C(=O)Nc2nc(C)c(Cl)nc2)cn2c(n1)CN(Cc1ccc(F)cc1Br)CC2 96051,CC(=O)CCCC(=O)N1CCCC1CNC(=O)C(c1cccc(Br)c1)(C)C 96052,C1(C(N2CC(CNC(=O)CCCCCO)C(C(F)(F)F)C2)=O)Cc2ccncc2C1 96053,Cc1nc2c(s1)CCCC2C(=O)NC1CC(NC(c2cccc3sncc23)=O)C1 96054,c1(C(N2CCCC(CNC(c3cncs3)=O)CC2)=O)c(F)ccc2c1OCO2 96055,N1(C(C(c2ccc(Cl)cc2)N(C)C)=O)CCC2C(NC(c3ccccc3F)=O)C12 96056,c1(C(=O)NC(CNC(c2cc(C)nn2C2CC2)=O)C2CC2)c(Cl)ccc(C)c1O 96057,C1(C(=O)NC2C=CCN(C(C3C(CC)CCO3)=O)C2)CC(=O)CC(=O)N1 96058,c1(C(=O)OC)ccc(C(=O)NC(CNC(c2ccn(CCOC)n2)=O)CO)s1 96059,N1(C(c2c(C)c[nH]n2)C(=O)NCCCF)CCN(c2cccnn2)CC1 96060,C1(O)(C(C)NC(=O)CC2CCOC2)CCN(C(C2COC3COCC23)=O)CC1 96061,c1(C(=O)NC2(CCOC)CCN(C(CC(=C)C)=O)C2)cn2cnnc2cn1 96062,C1(C(N(OC)C)=O)CC(O)CN1C(C)=O.C(C)(C)C 96063,CC(C(C)(C)CO)NC(c1n[nH]c(CO)n1)C 96064,N1(C(C(CCOC)C)=O)C2CCC1C(F)C(NC(c1c(C)coc1C(C)C)=O)C2 96065,c1(CNC(C)CC(=O)Nc2ccc(-c3nn[nH]n3)cc2)ccc2c(c1)C(=O)OC2 96066,N1(C(C(CC)O)=O)CCN(C(=O)CCN2CCCS2(=O)=O)C(CC(=O)NC)C1 96067,C1(NC(CCC2(C)CN(C(c3cc(COC)no3)=O)C2)=O)CCSC(C)C1 96068,N1(C(=O)Cn2cc(C3CC3)nn2)CCC2CN(C(=O)C(O)c3ccco3)CC2C1 96069,C1(C(C)NC(c2cc(C(C)(C)C)n[nH]2)=O)CCN(Cc2cc[nH]c2)CCC1(F)F 96070,c1(CNC(c2cccc(NC(c3cc(CC)n(C)n3)=O)c2)=O)nc(Cl)ccc1F 96071,c1(C(=O)NCCN(C(=O)CC2(N(C)C)CC2)CC)ccc(C(C)S(N)(=O)=O)cc1 96072,c1(C(N(CCN(C)CC2CCCC2)C)=O)cc(-c2ccoc2)on1 96073,Cc1cnc(C(=O)NC2CN(C(c3c(O)cccc3F)=O)CC2CO)c(C)c1 96074,c1(CN2CC(CNC(c3ncn(C)n3)=O)C2)ccc(F)cn1 96075,CC(C)C(C(C)NC(c1cscc1Br)=O)NC(c1ccc(CO)o1)=O 96076,C=CCCC(C)NC(=O)C(C)CN(C)C(c1csnc1OC)=O 96077,c1(NC)ccc(Cl)c(C(=O)NCC(C(C)(C)C)NC(=O)C(C)c2ccon2)c1 96078,C1(NC(C2CC(=O)NCC2)=O)CN(C(c2cnc(Cl)c(Cl)c2)=O)CCC1(F)F 96079,CCCS(=O)(=O)CC(=O)NC1CS(=O)(=O)CC1NC(=O)CCC(CF)CF 96080,C1(CC(=O)N(C2CCOC2)CCO)C2CCC(C2)N1C(=O)CC1CSC1 96081,C1(NC(C2CCC(F)CC2)=O)CCCC2CN(C(C3CCS(=O)(=O)CC3)=O)CC12 96082,C=CCC(CC(=O)NCc1cccc(C#N)n1)NC(=O)Cc1ccc(OC)cc1 96083,N#Cc1cc(NC(C2COCCN2C(C2CC2C2CC2)=O)=O)cc(Cl)c1 96084,C=CCC(C)(CNC(=O)C1=CCC(NC(=O)CCOC2CCCC2)C1)CO 96085,c1(OC)cc(OC)c(C(N2CC(C)(NC(=O)C(O)Cn3cncn3)C2)=O)c(N)c1 96086,c1(C(=O)NC2C(C)CCN(C(=O)CCOC3COC3)C2)cc2cccc(Cl)c2[nH]1 96087,c1(C(=O)NC2C(CNC(Cc3cc(C(C)C)on3)=O)CC2)cnc2c[nH]nc2c1 96088,N1(CC)CC2(CN(C(=O)C(C)N(CCOC)C(c3nc(=N)cc[nH]3)=O)C2)C1 96089,C1(CC)(CO)CCN(C(=O)C(CO)NC(c2cc(Cl)no2)=O)C1 96090,C=CC(C)(CCOC)C(=O)N1CCCC(NC(C23CCC(CC2)OC3)=O)C1 96091,Cc1cc(C2(C)C(=O)N2)ccc1Cl.C(CC(C)CO)N(C(=O)OC(C)(C)C)C 96092,c1(OC)ccc2[nH]nc(C(=O)NC(C)CNC(c3c(F)cc(C)cc3F)=O)c2c1 96093,C=Cc1cccc(CN2CCN(CCC(N3CCC(C)CC3)=O)CC2)c1 96094,CC1CN(C(c2cccn3ncnc23)=O)C(C)CN1C(c1ccc(O)nc1Cl)=O 96095,CCCC(CCC)CC(=O)NCC1(F)CC(CNC(=O)CC(CC)OC)C1 96096,C(CO)(CCCCNC(C1(CF)CCC1)=O)NC(=O)COc1ccccc1 96097,c1(C(=O)NC2CC3CN(C(c4ccc(F)cc4F)=O)CC23)cccc2nc[nH]c12 96098,C(=O)(C(C)CS(C)=O)NCC(C12CCC(CC1)C2)NC(c1sc(C)c(O)n1)=O 96099,c1(Cn2cc(NC(C3C(C(=O)OC)C3)=O)c(C#N)n2)cc2ccc(Cl)c(F)c2o1 96100,c1(C(=O)NCC2C3CN(C(CNC=O)=O)CC32)ccc2ncccc2c1F 96101,c1(CN=C(NCC(CC)(C)OC)NCC(C)(C)C)cc(S(C)(=O)=O)ccc1F 96102,C12COCCC1CC(=O)N2.CS(=O)(=O)SC1CC1c1ccco1 96103,C1(NC(C(CCC)O)=O)CCCN(C(=O)CCc2ccc(F)nc2)CC1 96104,C1(C(N2CCC(CN(C)CC)C2)=O)C2CC3C(C2NC(=O)C(O)C(F)(F)F)C13 96105,C(CC(=O)NC1CCn2ccnc2C1)(C(C)(C)C)NC(C(=CC1CCCC1)C)=O 96106,c1(-c2c(C)occ2)nc(CC2CCC(O)C2)n(C2CCC2)n1 96107,c1(C(=O)NC(CC=CC)C(=O)NCC=CC(C)(C)C)cnc2ccccn12 96108,C(=O)(C1=CCOCC1)NCC1(C)CCN(C(=O)CCC2CCCCC2)C1 96109,N1(C(C2C(C(N)=O)C2)=O)CC2CCC(C1)N2C(c1ccc(F)c(N)c1)=O 96110,CC1COCC(CNC(C2CC2c2cccnc2)=O)O1 96111,c1(NC(CC)CNc2ccccc2)nccc(=NC(C)c2cccnc2)[nH]1 96112,c1(OC)ccc(C(N2CC(NC(C3CCOCC3)=O)C3CC3C2)=O)cc1[N+](=O)[O-] 96113,c1(CCC(=O)NC2CC3CCC2N3C(C2CC3(CC3)CO2)=O)ccc(O)c(F)c1 96114,CC(C)C(C(=O)NC1(C(N)=O)CC1)n1cc(C(O)C(C)(C)C)nn1 96115,C1(NC(CCc2cc(C)sc2C)=O)CCCCN(C(C2(CF)CCC2)=O)C1 96116,c1(OC(CC2CCN(Cc3cn(CC)nn3)CC2)=O)ccc(C)cc1CC#N 96117,N1(C(C2CCN(C(c3cscc3Br)=O)C2)=O)CCC(O)(CO)CC1 96118,CCC(CN(C)C)CC(=O)NC1CC(CNC(=O)C(=O)Nc2ccccc2)C1 96119,c1(NC(=O)NC2CC2c2cc(F)ccc2F)ccc2c(F)n[nH]c2c1 96120,C(=O)(CC(C)P(C)(C)=O)NCCC(CNC(C1(n2cccn2)CC1)=O)OC 96121,C1(C(=O)NCCOC(CCOC)c2cccs2)(NC(CNC(C)=O)=O)CC(F)C1 96122,C1(COC)CCC(C2COCCN2C(=O)NCCC2CCSC2)O1 96123,N1(C(C(C=C)O)=O)Cc2ccccc2CC1CNC(c1cc(CC)on1)=O 96124,c1(C(=O)NCCC2CCN(C(CS(CC)=O)=O)C2)cc(F)cc(C)c1C 96125,C1(CC(=O)NC(CC)(C2CC2)C2CC2)CN(C(=O)CCCCOC)CCC1C 96126,N1(C(c2n[nH]c(C)c2O)=O)CC(=O)NCC1C(=O)NC1CCOC1(C)C 96127,C1(CNC(C(F)=CCC)=O)CN(C(c2ccc(N3CCCCC3)nc2)=O)CCO1 96128,CC(C)(C#N)CC(=O)NCCC1CCN(C(c2cn(CC(N)=O)nn2)=O)CC1 96129,C(=O)(CC(C)c1ccco1)NCCN(C1CCCCC1)C(CSCC#C)=O 96130,Cc1sc(Cl)c(C(=O)Nc2ccc(NC(=O)NC(C)CCCC(C)C)cc2)c1C 96131,C(=O)(C(C(C)C)C(C)C)N1CC(COC)(CNC(=O)CC2CC3C=CC2C3)C1 96132,C1(C(N(CCCCC2CCCC2)C)=O)CCCN1C(=O)C(=O)NC1CCCCO1 96133,N1(C(C2CCC(C)O2)=O)C(C(=O)N(C)CC2(C)CCC2)C2CC(O)C1C2 96134,C1(NC(c2c(SCC)cccn2)=O)CC2CC1CN(C(=O)CC1CC3CC3C1)C2 96135,C1(CC(=O)NC(CC(=O)OCC)C)CN(C(c2ncsc2C)=O)CCO1 96136,c1(C(=O)NCCN(CC(C)O)C(=O)CSc2nnnn2C)cccc2nsnc12 96137,c1(OC(C(=O)NC(CN(C(CCC)=O)C)C)(C)C)ccc([N+](=O)[O-])cc1 96138,c1(CCN(C(c2c(C)cc(CC)o2)=O)Cc2cccnc2)ccc(Cl)c(Cl)c1 96139,C1(NC(C(C)c2cccs2)=O)CCN(C(c2c[nH]c(C(F)(F)F)c2)=O)CC1F 96140,c1(NC(CCCNC(c2ccc(C#C)c(C)c2)=O)=O)ccc(O)cc1[N+](=O)[O-] 96141,C1N(C(=NCCCCCCS(N)(=O)=O)NCCC(C)C(F)F)CCC1C 96142,C1(CCC(=O)NC(C2(C(N(CCCOC)C)=O)CC2)C)CCC(=O)C1 96143,c1(C(=O)NCCC2(NC(COC(CC)(C)C)=O)CC2)cc2ccc(OC)nc2[nH]1 96144,N1(C(C2CCCCC2(F)F)=O)CCC(F)(F)C(NCc2cc(Br)c(Br)s2)C1 96145,C1(NC(C2(CC#C)CCCCC2)=O)COC2(C1)CN(C(=O)C(C)N1CC(C)C1)C2 96146,N1(C(c2ccc(Cl)cc2)=O)CCC(N=c2ccc3nnc(C4CC4)n3[nH]2)CC1 96147,N1(C(COCCC#C)=O)CC(CN(C(=O)C(CCC)N(C)C)CC)C(C)C1 96148,C1(C)(C(=O)NC2(CCCC(=O)NC(c3cnsc3)C)CCC2)CC(=O)N(C)C1 96149,C1(C(N(CC(O)CNC(c2coc(CO)c2)=O)C)=O)CC12CC(C)(C)C2 96150,N1(C(C2(CNC(c3c(C)snn3)=O)CC3(CC3)C2)=O)CC2CCC(C1)C2C#N 96151,c1(C(=O)NC2(C)CC(C)(C)C2)cnc2ccccc2c1 96152,C1(C)(CC)CC(NC(C23CC(CO)(C2)OC3C)=O)CN1C(=O)CSC(F)F 96153,C1(NC(c2ncccc2C(F)F)=O)CN(C(c2cnc(S)nc2)=O)CC1C1CC1 96154,C1(n2cc(C3CN(C(C4CC45CCC5)=O)C3)nn2)CCOCC1O 96155,c1(C(=O)NC2CC(NC(CCCOCCC)=O)C2)ccc(C(C)C)cc1O 96156,C1(C)(C(=O)NCC(CC)NC(C)=O)CCCN(C(c2cccc(C)c2)=O)C1 96157,N1(C(c2ncccc2Cl)=O)CCCC2(CC(NC(=O)C(F)(F)C3CC3)CO2)C1 96158,c1(-c2n(CCC)nc(-c3ccn(C)n3)n2)nc(C)n2c1CCCC2 96159,C(C(CCO)C(C)(C)C)NC(C(=O)NC1C(C)(C)C1)=O 96160,N1(C(=O)Nc2c(C)c(O)c(Br)cn2)CC2(COC(C)(C)C2)C1 96161,c1(NCC2(CCOC)CC2)nc[nH]c(=NCC2Cc3ccccc3C2)c1C 96162,Cn1cc(Cl)c(C(=O)NC2CC2CNC(c2cnc(-c3ncccn3)s2)=O)n1 96163,C1(NC(C2(C(=O)OC)C(=C)CC2)=O)CCN(C(=O)CCc2nc[nH]n2)CC1 96164,C1(C(C)CNC(C2C=CCS2)=O)CCN(C(c2cnc(O)o2)=O)CC1 96165,c1(OC)nccc(C(N2CCCCC2CNC(c2cc[nH]c2C2CCC2)=O)=O)n1 96166,N1(C(CC(CCCC)O)=O)CC2(CCN(C(c3cc(C)nc(O)c3)=O)CC2)C1 96167,C1(C)(CC(=O)NCC2(CSC)CC2)CCN(C(C2C3CCC(=O)C23)=O)C1 96168,C1(F)(C(=O)NCC2N(C(c3c(CC)nco3)=O)CC=C2)CCCN(C)C1 96169,c1(-c2nc(C(C3CC3)OC)nn2-c2nc(Br)nn2C)cnn2c(C)ccnc12 96170,Cn1cc(C(N2CCC(F)(CNC(=O)CS(N)(=O)=O)C2)=O)c(Cl)n1 96171,N1(C(C2C(NC(=O)C(=O)C3CC3)CCC2)=O)CCC(C)(CO)C(O)C1 96172,C#CCCC(O)CCNC(c1cccnc1CNC(=O)C(C)C1(O)CCC1)=O 96173,C1(C(N2CC(SC)C(n3cc(C(C)(C)CO)nn3)C2)=O)CCCCN1N=O 96174,Cc1cnc2nccc(C(N3CC(CNC(c4cscn4)=O)CCC3C)=O)c2c1 96175,c1(NC(C2C(NCc3ccc(OCC)c(C#N)c3)C2)=O)nccc2scc(Br)c12 96176,N1(C(Cc2cc(C)[nH]n2)=O)CCC2CN(C(c3coc4c3COC4)=O)CC2C1 96177,N1(C(C)=O)CCN(C(=NC2CC2)NCc2noc(C(C)C)n2)CC1(C)C 96178,C(=O)(C(O)P(C)(C)=O)N1CC2C(C(N3C(C)(C(=O)OC)CC3)=O)C2C1 96179,C1(NC(c2c(NC)snc2C)=O)CCCN(C(=O)C(C)CC(C)C)CC1 96180,c1(C(N2CCC(C(=O)NCCCOC)(CO)C2)=O)cc(C#N)[nH]c1C 96181,C1(C(=O)NC(c2cnn[nH]2)C)CC(O)CN1C(C1CN(C(N)=O)C1)=O 96182,c1(CC(=O)NC(CNC(c2ncn(C)c2)=O)C2CC2)cccc(Br)c1 96183,c1(CC)ccc(CC(=O)NC2CCC(C)N(C(c3[nH]ccc3C)=O)C2)cc1F 96184,C(=O)(C1=NOCC1)N(C1CCCC(N(C)C(c2cncc(N)n2)=O)C1)C 96185,C(=O)(C#CC1CCCOC1)N1CC(CNC(CCC=C)=O)OC(C)(C)C1 96186,Cc1ccc(CN(CCO)C(c2c[nH]cc2Br)=O)cc1 96187,c1(C(=O)OCC)cc(C(N2CCCC2CCNC(=O)C(C)C2CCC2)=O)[nH]c1C 96188,C1(NC(C(F)OC)=O)CN(C(=O)Cc2cncn2C2CC2)CC1O 96189,c1(C(N2CCC(CSC)C2)C(=O)Nc2cccc(Br)c2)cc(C#N)ccc1F 96190,c1(CC)ccc(CC(=O)NC2CN(C(=O)CC(CC)OC)CC23CC3)c(OC)c1 96191,N1(C(CCCC)=O)CC2CCC(CNC(=O)CCc3cccc(F)c3)(C2)C1 96192,Cc1ccc(C(=O)N(C2CCN(C(c3cc(Cl)no3)=O)CC2C)C)nc1O 96193,CCC(F)(C(=O)OC)C(=O)N1CC(O)(C(C)NC(C2CN(S(=O)(=O)CC)C2)=O)C1 96194,CC1CN(C(=O)C=Cc2cn[nH]c2)CC(C)CN1C(c1cc(O)cs1)=O 96195,Cn1ccc(C(=O)NC2CC2C(=O)Nc2ccc(C(N)=O)cc2F)cc1=O 96196,C1(CCC)CCCN(C(=O)C(CNC(=O)C(C)(C)C2CC2)CCC)CC1 96197,C12(CNC(C3CC(CC)(CC)C3)=O)CCCC(CN1C(c1cncc(C)c1)=O)C2 96198,c1(NC(C2CCCC(C(=O)OC)C2)=O)nn(C)c2ccccc12 96199,c1(OCCC)ccc(NC(C2CN3CCC2C3)=O)c(OC)c1 96200,C1(CNC(c2cc(Br)c[nH]2)=O)CCN(C(C23CCCC2C3(F)F)=O)C12CC2 96201,C1(C(=O)N(C)CCC2CCCO2)(CC)CN(C(=O)CN2CCOCC2)C1 96202,C1(CC(=O)NCC(C(C)C)NC(C2CCC(C(=O)OC)C2)=O)CCCC(C)(C)O1 96203,C(CC(C)C)(C(=O)NCC(O)C(C)(C)O)NC(C1C(COC)CC1)=O 96204,C=CCC(F)(F)C(=O)NC1CN(C(c2cc(CC)ccn2)=O)CC1OC 96205,N1(C(c2cnc(CC)s2)=O)CCCCC(NC(c2c(NC(C)=O)c[nH]c2C)=O)C1 96206,CC1CN(C(c2ccnn2CCF)=O)CCC1CNC(C1CC2(CCOC2)C1)=O 96207,CC1CN(CC(=O)NCC2(O)CC2)CCC1NC(c1cn(CCC2CC2)nn1)=O 96208,Cn1ccc2ccc(C(=O)NC(C)(CNC(=O)CCN3CCCCC3)CO)cc12 96209,c1(C(C(=O)NCCC)N(CCC(C)OCC)C)ccc(C)c(OC)n1 96210,N1(C(CS(c2cccc(C)c2)=O)=O)CC(S(=O)(=O)C2CCCCC2)C1 96211,N1(C(C2N(CC)CCOC2)=O)CCCC(O)(CCNC(=O)Cc2ncoc2C)C1 96212,Cc1nn(-c2ccccc2)nc1CC(N1CC(Cn2cc(C3CC3)nn2)C1)=O 96213,C(C(C)C(F)C(=O)NC(CO)C(F)(F)F)NC(c1cccc(C)c1)=O 96214,c1(C(N2CCC(CC(N3CCC(CC(=O)OC)CC3)=O)C2)=O)ccc(C#N)c(Cl)c1 96215,C(CCC(C)CC(=O)NC1(CF)CCN(C(=O)CN(C)CCO)C1)=C(C)C 96216,n1(CC(N2CC(NC(C3(C=C)CCC3)=O)C3(C2)CC3)=O)nc2n(c1=O)CCCC2 96217,CC(C)CCC(=O)N(CC(O)CN(CC(=O)NS(=O)(=O)Cc1ccon1)C)C 96218,C1(NCCC2CC=CCC2)COC2(CCC2)C1 96219,N=c1c(C(=O)OC2CCCC2(F)F)c[nH]n1-c1ccc(Cl)cc1 96220,N1(C(C(c2cncnc2)C)=O)C2CCC1C1CC1(NC(=O)C=C1CCC1)C2 96221,C(=O)(C(C)(C)C(=O)N1CCCCC1CNC(C1(C2CCCO2)CC1)=O)NC 96222,Cc1ccc(CC(N2CCC(C(F)F)(CNC(C3CCC3(C)C)=O)C2)=O)c(C)c1 96223,C(=O)(CC(F)(F)F)NCC(=O)N(C)CC1N(C(c2nnc(CC)s2)=O)CCC1 96224,c1(C(N2CCCCC(CNC(C3C(C)C3)=O)C2)=O)ccc2nn[nH]c2c1 96225,Cc1ncc(Br)c(C(N2CCSC(C(N3CCCC(F)C3)=O)C2)=O)n1 96226,CC(C)(CCNC(c1csc(-c2ccccc2)c1)=O)C1CC1 96227,C(=O)(C1=C(C#N)CCC1)NCCCC(C)(C)NC(C1C(CC)OCC1)=O 96228,CC1SCCCN1C(N1CCCC1c1cccnc1)=O 96229,C1(C(N(CCC(=O)NCC2C3COCC23)C)=O)OC2CCC1C2 96230,CC1CC(NC(c2ncccc2CO)=O)CN1C(=O)CCc1cscn1 96231,N1(C(COC(C)C)=O)CCCC(NC(c2ccn(C)c(=O)c2)=O)C(F)C1 96232,N1(C(CC2(C=C)CN(C(c3cc(OC)no3)=O)C2)=O)CC2(C1)CC2(F)F 96233,c1(OCC)ccc(CCC(=O)NC(C)(C)C(C)NC(=O)C=Cc2ncco2)cc1 96234,C1(CC(O)CO)(NC(=O)NCc2cc(-c3ccccn3)no2)CCCNC1 96235,N1(C(c2c(C)cno2)=O)CCN(c2nc(C(C)C)ns2)C(CCO)C1 96236,c1(C(=O)NCN(CC)Cc2cn(C)nn2)cc(F)n(C)n1 96237,C1(C)(C(=O)NCCCN(C(C)=O)C)CCN(C(C2CC(=C3CC3)C2)=O)CC1 96238,c1nc(CC)sc1CC.c1(CC)cn(NCC2CC2)nn1.C12CC(C1)C(=O)N2 96239,C1(C(C)(C)C)CCC1C(N1CC(C(O)C(=O)NCc2cnc[nH]2)C1)=O 96240,N1(CC)CCC(NC(C2(CCNC(=O)Cc3ccc(C)o3)CC2)=O)C(C)C1 96241,N1(C(C2(CC=C)CC2)=O)CCCC(C2(NC(c3cnc(Cl)c(F)c3N)=O)CC2)C1 96242,c1(NC2CCN(C(=O)NC)CC2)nc(C(F)(F)F)ccc1I 96243,c1(OC)ccncc1C(=O)NC(c1nocc1C(=O)N(C1CC1(C)C)C)C 96244,CC(C)CC(C)(O)C(=O)N1C2CCC(C(=O)NCc3cnns3)C1CC2 96245,N1(C(c2ccc(SC)o2)=O)CCC2(NC(c3cc(=O)n(C)cn3)=O)CCCCC12 96246,c1(OC)cc(C=C(C)CN2CCC(O)CC2C(=O)N(C)C)c(OC)cc1C 96247,N1(C(CC(COC)(C)C)=O)CCC(N=[N+]=[N-])(C(=O)NOCC(N)=O)C1 96248,Cn1ccc2[nH]c(C(N3CCC(NC(C4(C5CCC5)CC4)=O)C3(C)C)=O)cc12 96249,c1(CNC(CC2N(C)CCC2)=O)ccc(C(=O)NCC(N2CCCC2)C)nc1 96250,C(C(=O)N=c1cc(C)n(C2CC2)[nH]1)=C1CN(C(C2C(OC)CC2)=O)C1 96251,N1(C(COC)=O)CCC2(CCCN2C(=O)CCc2ccc(OC(F)F)cc2)C1 96252,Cc1cccnc1CC(N1CCC(C(F)F)(CNC(c2cc(CF)on2)=O)C1)=O 96253,c1(C(N2CC3C(CNC(C=COCC)=O)(C3)C2)=O)cc(Cl)cc(Cl)c1OC 96254,CC1(C(N2CCCC2c2cn(-c3ccc(CN(C)C)cc3)nn2)=O)CCCC1(F)F 96255,c1(C(=O)NC(CNC(=O)C=CCn2cncn2)CO)ccc(-n2ccnc2)nc1 96256,CN1CCC(CNC(C(C)(C)CCCC)(c2nnnn2-c2ccccc2)C)C1=O 96257,c1(NC(C(C)NC(=O)NC)=O)cc(NC2CCCC2)c(F)cc1F 96258,Cc1nc(NCC(F)C2CCC2)cc(=NC(C)c2ccc(NS(C)(=O)=O)cc2)[nH]1 96259,c1(NC(C2CC2NCc2cscn2)=O)cccc(Cl)c1I 96260,c1(Cc2ccccc2)nc2c(s1)C(NCc1cnn(C3CC3)c1)CCC2 96261,N1(C(COCCOC)=O)CCC2(CNC(=O)C3=NNC(=O)CC3)CCCCC12 96262,c1(NCC(C)CNC(=O)CC2CC(O)C23CCC3)ncnc(N(C)C)c1[N+](=O)[O-] 96263,c1(CN2CCCC(C(N3CCOC4CC34)=O)C2)cnc(Cl)cc1Cl 96264,c1(C(=O)NC2(CN(C)C(c3ccc(C(C)(F)F)cc3)=O)CC2)cccc(N(C)C)n1 96265,Cc1c(C(N2CC(C)(NC(C3OC4CCC3C4)=O)C2)=O)[nH]c2c(Cl)cccc12 96266,c1(CNCC2CN(C(C(C)NC(c3ccoc3)=O)=O)CC2C)cccc(Cl)c1F 96267,N1(C(CCCCC=CC)=O)CCC(C2(NC(=O)Cc3sccc3C)CC2)C1 96268,c1(OC)cc(NCc2c(C(N)=O)cnn2-c2ccccc2Cl)ccc1O 96269,c1(SC)nn(C)cc1C(N1CCC(C)C1CNC(C1(C(F)F)CCC1)=O)=O 96270,N1(C(c2cnn(C)c2C2CC2)=O)CCC2(CCN(C(=O)CC3(C)CC3(Cl)Cl)C2)C1 96271,c1(C(=O)NCC(CN(C(c2c(O)ccc(CC)c2)=O)C)C)cc(S(N)(=O)=O)co1 96272,c1(OC)cc(NC(c2cccc(F)c2Br)c2nnnn2C)cc(Br)c1OC(F)F 96273,C1(OC)CCC(C(=O)NCC2CCCCC2NC(c2cc(C(F)F)cs2)=O)CC1 96274,Cc1ccc(Cl)c(N)c1C(N1CCC(CNC(=O)C(C)(F)F)C(F)(F)C1)=O 96275,C=CCCC(C(=O)N(CCNC(=O)CC(=O)NC1CCC1)CC)c1ccccc1 96276,C1(CNC(C(C)(C)C#N)=O)CCCCN(C(C2SCCCS2)=O)C1 96277,c1(C(=O)OC(c2ccc(F)cc2F)C(=O)OC)cccc2nsnc12 96278,C1(CNC(=O)N(C2CC2)Cc2cc([N+](=O)[O-])cs2)(CO)CC2CCC1CC2 96279,CCC(C)(O)C(=O)NC(C)CNC(c1cnn(Cc2ccccc2)c1Br)=O 96280,C1(NC(c2cnn(C)c2F)=O)CCC2CC1CN2C(c1cc([N+](=O)[O-])c[nH]1)=O 96281,c1(CSCC(=O)NCCNC(C2ON=C(CC)C2)=O)n[nH]c2ccc(Cl)cc12 96282,Cc1cc(NC(C2CCCCCN2C(c2cccs2)=O)=O)ccc1O 96283,CCCCCCCCN(C(=O)C(CC1CC1)N(C(=O)C(C)OC)CC)CC 96284,C1(C(N2CC(CC)N(C(c3cnn(C)c3)=O)CC2)=O)COc2cc(F)ccc2C1 96285,N1(C(c2c(OC)c(Br)ccc2)=O)CCn2cnc(C3=CCSCC3)c2C1 96286,Cc1cc(C(=O)NCCN2CCN(C(C3CCNC3=O)=O)CC2)cnc1O 96287,N1(C(COCCC)=O)CCCC2(CCN(c3ccc([N+](=O)[O-])c(OC)c3)C2)C1 96288,CCC(C)(CC)C(=O)NCCCCC(C)NC(C1CCCC(C)CC1)=O 96289,C(=O)(C(F)(F)C(F)(F)F)NCC(CC=C)NC(c1conc1-c1ccccc1)=O 96290,C1(C)(CC)C=C(C(=O)N2CC3(CNC(c4cc(OC)cc(F)c4)=O)CC2CO3)C1 96291,CC(C)CN=C(NCC1CCN(C(C)C)C1)N1CCCC2(CCCNC2=O)C1 96292,CCC(CC(C)C)C(=O)NCC1CC2(CC2)CN1C(c1cn(CCOC)nn1)=O 96293,CS(=O)(=O)c1ccc(C(N2CCC(N(CCO)C(C3CCNC3=O)=O)C2)=O)cc1 96294,C1(CNC(CC(C)N(C)C)=O)CN(C(c2n[nH]c3c2COCC3)=O)CC(C)(C)O1 96295,CCCC(C(C(=O)NC)N1CC(O)C2(CCC2)C1)OC 96296,c1(CC(N2CC(=C(CNC(C(CC)SC)=O)F)C2)=O)ccc(F)cc1C 96297,C(=O)(C(F)(F)C(F)(F)F)NC1CCC(CNC(C2CC(OC)CN2C(C)=O)=O)C1 96298,N1(C(C=CC(CC)C)=O)CC(O)(C(F)C(=O)N2CC(OC(=O)N(C)C)C2)C1 96299,N1(C(C2CC=C(C)CC2)=O)CC2(CCCC2NC(C2(C3CCC3)CC2(F)F)=O)C1 96300,c1(NC(c2nc(C(N3CCC34CCCCC4)=O)cs2)=O)c(F)cc(F)cc1Cl 96301,C1(CN(C(=O)C(C)(O)COC)CC)CCN(C(c2cnn(C)c2SC)=O)CC1 96302,N1(C(C2(C)CC(=C)C2)=O)CCN(C(c2cnc(C)o2)=O)C(c2cn[nH]c2)C1 96303,CC(C(=O)N1CCC(n2cc(-c3ccccc3O)nn2)CC1)C(F)F 96304,N1(C(=O)Cn2nnc(=O)[nH]2)CC2(CCN(C(c3ccc(Br)cc3F)=O)CC2)C1 96305,N1(C(C(Cn2ccc(C)n2)C)=O)CC2CN(C(c3ccc(C)c(O)c3)=O)CCC12 96306,N1(C(CC(COC)(C)C)=O)CCCC2(NC(C3CCCCNC3=O)=O)CCCC12 96307,c1(C(N2CC=CC(NC(COCC(C)C)=O)C2)=O)cn2ccncc2n1 96308,N1(C(CNC(c2cc(COC)no2)=O)=O)CCC2(CC(NC(C3CCOCO3)=O)C2)C1 96309,c1(OCC(=O)N(CC(C)O)CCNC(=O)CNC=O)ccc(Cl)cc1 96310,c1(C(N2C(CNC(CCOC(CC(C)C)C)=O)CC2)=O)ccc([N+](=O)[O-])s1 96311,c1(C(=O)NC(CN2CC(C)CC(C)C2)C)nc(Cl)c(Br)cc1[N+](=O)[O-] 96312,c1(C(=O)O)n[nH]c2cc(C(=O)Nc3ccc(=NCc4cc(Br)co4)[nH]c3)ccc12 96313,N#Cc1ccc(F)cc1CNC1CCN(c2ncccn2)C1 96314,CC1C(NC(=O)CC2=CCN(C)CC2)CC2CCC1N2C(C1CCCOC1C)=O 96315,C12(CNC(c3cccc(C)n3)=O)CCCCC1N(C(c1ccc(O)cc1)=O)CC2 96316,c1(NC(C)=O)cc(Cl)ccc1S(=O)(=O)Nc1ccc(C(C)(C)S(C)(=O)=O)cc1 96317,C(N=c1[nH]c(=N)[nH]c(=NCC(CSC)N2CCN(CC)CC2)[nH]1)C1(OC)CCC1 96318,c1(OC)ccccc1CC(=O)C(=O)NCC1CCCN1C(C1CCOCC1)=O 96319,CCCS(=O)(=O)CC(=O)NC1CC2(C1)CN(C(=O)C(C)(C)C1CCOCC1)C2 96320,C1(C(=O)NCC2(NC(CCC3C(C)(C)C3)=O)CCOC2)CC(=O)CC(=O)C1 96321,c1(C(=O)NC(CNC(c2c(C(C)C)c[nH]n2)=O)(C)C)ccc2c(c1)C(C)C(C)O2 96322,C1(CNC(CC2(CSC)CC2)=O)CC12CCN(C(c1c(C)nsc1Cl)=O)CC2 96323,CN1CCOCC1CNC(C1(NC(C2CCCOCC2)=O)CCCCC1)=O 96324,C1(C(=O)NCC(C)NC(c2cnoc2C2CCC2)=O)CCCCC1O 96325,N(C(=NCCOC(F)(F)F)NCC(Cc1ccoc1)CO)C1C(C)C1 96326,c1(C(=O)NNC(=O)C2CC(O)CN2Cc2cccnc2)cc(F)cnc1Br 96327,C1(C(=O)NCC(C)NC(c2c(CCC)n[nH]c2)=O)CC12CCC1(CC1)CC2 96328,Cc1cc(C(N2CC(F)(C(N3CCCC(CC(C)C)C3)=O)C2)=O)nc(C)n1 96329,c1(C(=O)NC(CCOC)CNC(=O)C(C)NC(=O)C(C)(C)C)ccc(N)c(F)c1 96330,CC(F)(CC1CCCC1)C(=O)N1CCC1CNC(c1cc(Cl)cs1)=O 96331,N(C(=NCC(C)C)N1CCN(Cc2ncoc2C)CC1)C(COC)C 96332,C1(CNC(C(C2CCN(C(CCOC(C)C)=O)C2)C)=O)C2CCCCCC12 96333,C1(C(=O)NCCN(C(Cn2c(C)ccn2)=O)C2CC2)CCC(C(F)(F)F)CC1 96334,CC(CC(N)=O)C(=O)NC(CC(N)=O)C(=O)NC(C)CCO 96335,N1(C(CC=C=C)=O)CCN(C(=O)C=Cc2ccc(-c3ccccc3)s2)C(CO)C1 96336,c1(N2CCC(N(C)C(C3CC4CC4C3)=O)C2)nccc(C#N)c1[N+](=O)[O-] 96337,C1(c2cn(CC3N(C(C(c4cn(C)nc4)O)=O)CC3)nn2)CC2C=CC1C2 96338,C1(C(=O)Nc2c(COC)nn(C)c2)N(C(C2CC=C(C)CC2)=O)CCC1(C)C 96339,N1(C(CCSCCC)=O)CCC2(CCN(C(=O)CC3CCCN3C)CC2)C(C)C1 96340,c1(NC(CC)CO)ccc(S(=O)(=O)NC2(C3CC3)CCOCC2)cc1F 96341,c1(C(=O)Nc2ccc(CN(C)CC)cc2)cc(Br)cc(Cl)c1Cl 96342,C1(C)(C(N2CC=CC(C(=O)NC(CCC(C)C)C)C2)=O)CCC2CC2C1 96343,c1(OC(C)C(=O)OCC2CONC2=O)cccc(Br)c1 96344,N1(C(C2CCCN(C)C2)=O)CC(CNC(c2c[nH]c(=O)cn2)=O)C(C)(C)C1 96345,c1(CONC(c2cn(C)nc2CCC(F)(F)F)=O)c(F)cccc1I 96346,C1(C(N2C(C(=O)NC3(C)CC(O)(CO)C3)C=CC2)=O)CN2CCN1CC2 96347,N1(C(CCC(=O)NC)=O)CC(C)CN(C(c2cc(CO)ccn2)=O)C(C)C1 96348,C(c1csc(C)n1)=CC(=O)NC(CCNC(c1n(CC)cnn1)=O)C 96349,c1(OC)cncc(CCC(=O)NCC(C2CCC2)NC(=O)C=C(C)C(F)F)c1 96350,c1(C(C(=O)NCCOCC)N(CCC(=O)OC)CCCOC)cc(Cl)sc1Cl 96351,c1(CCn2cc(CNC(CCCOC(CCC)=O)=O)nn2)cccnc1C 96352,N1(C(=O)OC(C)(C)C)CC(N=[N+]=[N-])CC1C(=O)NCC1(C(F)(F)F)CCC1 96353,C1(CCNC(c2c(CC)ccs2)=O)CN(C(C2CC(F)C(=O)N2)=O)CC1C 96354,c1(C(=O)NC2CCCN(C(c3cc(C(CC)C)no3)=O)C2)c(C)ccc(C)c1N 96355,c1(C(=O)NC(CNC(CSCC#C)=O)CCOC)cnc2c(C)cccc2c1 96356,CC(CCNCCc1ccnc(Cl)c1F)P(C)(C)=O 96357,N1(C(COC(C)(C)C)=O)CC(C)(C)OC2(C1)CN(C(C1C3CS(=O)(=O)CC13)=O)C2 96358,C1(C)(C(N(CC(C)O)CCNC(=O)Cc2ccno2)=O)CCC(=O)N1 96359,c1(CC)nc(CCNC(C2CC(C)N2C(c2ccnn2CCF)=O)=O)n[nH]1 96360,N1(C(=O)CCSC2CCCC2)CC2(CCN2C(c2ccccc2C(F)F)=O)C1 96361,C(c1scnc1C)=CC(=O)N(CC(C)(C)NC(c1c(CCC)occ1)=O)C 96362,c1(C(=O)NC2C(NC(c3cc(Cl)cs3)=O)COCC2)ccc(F)c2c1CCC2 96363,C(=O)(CC1=CCOCC1)N1CCC(O)(C(C)NC(=O)Cc2c[nH]nc2O)C1 96364,Nc1ccc(C(=O)NCC2CCN(C(C3CC(F)C(=O)N3)=O)C2)cc1F 96365,C1(CC(=O)NC2C(NC(c3c(OC)nsc3)=O)CCOC2)SC2=NCCN2C1=O 96366,n1(CC(=O)NC(C)CC(C)NC(=O)CSCC(F)(F)F)nc2n(c1=O)CCOC2 96367,CC1CC=C(C(=O)NC(C2CCCC2)CNC(=O)CSC(C)(C)C)CC1 96368,Cc1ncc2cc(C(N3CCC(c4nc(C5CC5)no4)CC3)=O)c(O)nc2n1 96369,c1(COC)nn[nH]c1C(=O)NCCC(C)N(C)C(C1(OC)CC1)=O 96370,CCC(C)CCCCC(=O)N1CCC(NC(c2cnc(N(C)C)cn2)=O)CC1C 96371,N1(C(C2CC(CC)C2)=O)CCN(C(C23C4C5C2C2C3C4C52C)=O)CC(O)C1 96372,c1(CC(N2C(CNC(C3OC4CCC3C4)=O)CC(F)C2)=O)nc([N+](=O)[O-])n[nH]1 96373,C1(C(=O)NCC(CC)(C)NC(=O)CN(C)CCOC)OCC2COCCC12 96374,Cc1nc(C(C)C)nc(O)c1C(=O)NC1CCC(NC(c2cnc[nH]2)=O)C1 96375,C1(CCNC(COCCN(C)C)=O)CN(C(=O)Cc2cncnc2)CCO1 96376,C1(NC(CCCN(C(=O)CCC(F)(F)F)C)=O)CC2CCC(C1)N2C 96377,C1(C2CCOCC2)(C(N2CC3(CN(C(C4CC4F)=O)C3)OCC2)=O)CCOCC1 96378,CC1CCc2onc(C(=O)NCCC3CCN(C(c4ccc(Cl)cn4)=O)C3)c2C1 96379,C1C(C(C)C)N=C2C=CN=C(N2)NC(=O)C(C)O1.C(COCCOCCOC)OC 96380,c1(NC(=O)Nc2ccccc2Br)cncc(-c2ccc(N3CCOCC3)nc2)c1 96381,C=CCCC(C(=O)NCC=Cc1ccccc1)NC(C1CC2(CC2)C1)=O 96382,C#CCC(C)(C)C(=O)N1CC(C(N2CC(C(F)(F)F)C2)=O)C2(CC2)C1 96383,C1(CC=C)(NC(COCCC=C)=O)CN(C(c2cc(Br)cs2)=O)C1 96384,C(C(C)N(C)N1CCCC1C1CCCCN1C1CCC1)c1c(C)cccc1 96385,O(N=c1cc[nH]c2ccc(-c3cnc(N)c(Br)c3)cc12)C(C(=O)OC)C 96386,c1(CC(N2C(c3cn(CC(CC)C)nn3)C(C)CC2)=O)ccc(F)c(OC)c1F 96387,c1(NC(C)CCNC(C2CC2(F)F)=O)nnccc1C#N 96388,N1(C(C(C)OCC)=O)CC(C)C(C)(CNC(c2ccnn2CC(F)F)=O)C1 96389,c1(C(=O)NC2CC(NC(CCc3c(OC)cccc3)=O)C2)nc(Cl)ccc1N 96390,N1(C(C(c2cccc(Cl)c2)C)=O)CC2CC(C1)N(C(=O)C(O)CCN(C)C)C2 96391,N1(C(C(=O)N(C(C)C)C)C)CCC(NC(c2ccsc2C(F)F)=O)C(C)C1 96392,C1(C(=O)NC2CC(C(C)C)OC2)CN(C(C2(C)CC(=O)C2)=O)CC1F 96393,C1(C(=O)NC23CC(NC(C(C)c4ccco4)=O)(C2)C3)CN2CCN1CC2.C12CC1C2 96394,Cc1nc2cc(C(N3CCC(NC(=O)C4=CCCOC4)C(C)(C)C3)=O)cnc2[nH]1 96395,C1(NC(C(COC)O)=O)CC2CC(NC(c3cnccc3C(=O)OC)=O)CC2C1 96396,O=C(NNC(=O)C12CCC1C2)C1CCC1 96397,CC(C)CCCC(C)C(=O)NCC1CN(C(c2ccc(CO)o2)=O)CCCO1 96398,N1(C(c2c(C)ccs2)=O)CC2CN(C(=O)CC3COCCN3C)CC2(C)C1 96399,c1(C(N2CCCC(C)(NC(c3cc(C(N)=O)[nH]n3)=O)C2)=O)cc(F)c(F)c(F)c1 96400,C12(NC(C3CCS3(=O)=O)=O)CCCN(C(c3cc4ccsc4s3)=O)CC1C2 96401,c1(C(=O)NCC2C(CNC(C(=Cc3cnc[nH]3)C)=O)C2)nc2ccccn2c1F 96402,C1(NC(C2(COC)CC2)=O)CC(O)CN(C(c2c(OC)ccnc2O)=O)C1 96403,CCCC(C(=O)N(C)CCNC(=O)C=CC1CCCO1)S(N)(=O)=O 96404,C(=O)(CC(C)C(C)C)N1CC(CCCCNC(CCc2cnc(C)o2)=O)C1 96405,C(CC(C)C)(C(N)=O)NC(c1n(CC=C)nnn1)c1cnc(-c2ccccc2)s1 96406,CC(C)CC(CC(=O)NC(C(N)=O)C1CC1)NC(C1COCCC1C)=O 96407,C(=O)(CCC(=O)c1cccnc1)NCC(C)(C)CNC(c1ccsc1)=O 96408,CC(C)(C#N)C(=O)NCCCOCCCNC(C1CC(O)(c2ccccc2)C1)=O 96409,N1(C(CCCC(=C)C)=O)CC2(CCN(C(=O)C(C(C)(C)C)N(C)C)CC2)CC1C 96410,C1(F)(CNC(c2ccc(Oc3cccnc3)cc2)=O)CCN(C(=O)C2CC2)C1 96411,C1(CNC(CCCN(C)C)=O)CCCCN(C(=O)CC2(C3CC3)CC2)C1 96412,N1(C(COCc2onc(CC)n2)=O)CCOC(CNC(C2COCCN2C)=O)C1 96413,C1(NC(CCC(C)C)=O)CN(C(C2CCCN(S(C)(=O)=O)C2)=O)CCC1C 96414,c1(C(=O)NCC2(NC(=O)C=CI)CCCCC2)ccc2nc(O)[nH]c2c1 96415,c1(C(=O)NC2C(OC)CN(C(c3ccc(C)nc3O)=O)C2)ccc(N)c(O)c1 96416,C1(NC(CCCNC(N)=O)=O)CCCC(CNC(C2(N3CCOCC3)CC2)=O)C1 96417,C(=O)(C1CCCc2nn[nH]c21)NCCC1CC(NC(=O)C=CCF)C1 96418,C(=O)(NNC1(C)CCS(=O)(=O)C1)NC(CSc1ccc(SC)cc1)C 96419,N1(C(C2C(C)(C(=O)OCC)C2)=O)C2CCC1CN(C(c1cncnc1C)=O)C2 96420,N1(C(c2n(CC)ncc2C)=O)CC(CCNC(=O)CNS(C)(=O)=O)OC(C)C1 96421,C1(N(C(=O)CCC2CCC(=O)C2)C)CCCN(C(=O)CN2C(=O)CNC2=O)CC1 96422,C1(C(=O)NCCCc2ccsc2)CCCCN(C(c2ccc(O)nn2)=O)C1 96423,C1(C2CCC2)(C(=O)NCC2C(NC(c3cccc(C(F)F)n3)=O)CC2)CC1 96424,c1(C(=O)NC2C(CNC(C(C=C)O)=O)CC2)sc2ccc(C(=O)OC)cc2c1C 96425,C1(CCNC(C2(C(CC)(F)F)CC2)=O)(NC(c2cnc(OC)s2)=O)CCCC1 96426,c1(OC)ccc(F)cc1C(=O)NC1CC(C)N(C(c2cnc(N(C)C)s2)=O)C1 96427,Cc1cccc2[nH]c(C(=O)NCC3CCCCN3C(C3(C)CCCS3)=O)cc12 96428,C1(NC(C2C=CCC2)=O)CC2CC(C1)N(c1nccc(CO)n1)C2 96429,C(c1nc2ccccc2s1)=CC(=O)OCC(c1c(C(=O)OC)scc1)=O 96430,C1(NC(c2c(C)nn(CCO)c2)=O)CCN(C(=O)CS(=O)(=O)N(C)C)C12CCC2 96431,N1(C(c2cc3cc(Cl)ccc3o2)C(=O)NCCOC)CCOc2ccccc2C1 96432,Cc1nn2c(c1CNc1ccco1)CN(C(C1(n3nccn3)CC1)=O)CC2 96433,N1(C(c2ccc(OC)c(C)c2)C(=O)NC2CCCC2)CCC2(CC(=O)N(C)C2)C1 96434,c1(OC)ccc(CC(N2CCCC2CC(N2CCC(F)C2)=O)=O)c(OC)c1 96435,Cc1cc(C(=O)NC2CCN(Cc3cncc(C(F)(F)F)c3)C2)c(F)c(Br)c1 96436,N1(C(c2c(C)c[nH]n2)=O)CC(NC(=O)CC2CC23CC3)CC1(C)C 96437,CC1CCC(C(C)(O)CNC(=O)NCCNC(c2cnnn2C)=O)CC1 96438,c1(C(N2CCC(NC(c3cc(Cl)cc(F)c3F)=O)C2)=O)cccc2cc[nH]c12 96439,CC1=C(C(=O)NC(C)CN(C(=O)C(C)N(CC(F)(F)F)C)C)S(=O)(=O)CCO1 96440,C1(CN(C)C(N)=O)CCCN(C(C2CCCN2C(C2C3(CC3)C23CC3)=O)=O)C1 96441,C1(OC)CCC2(C(=O)NCC(C3CCCC3)NC(c3scnc3Cl)=O)CCC12 96442,C(=O)(C1COc2ccc(F)cc21)OCc1c2nnc(C)n2nc(Cl)c1 96443,c1(N(C)C(c2ccc(-c3cccc4cc[nH]c34)cc2)=O)nc2c(s1)CCCCC2 96444,S(=O)(=O)(c1ccc(Cl)cc1F)NC1C2CN(C(C3CC(=C)C3)=O)C(C2)C1 96445,c1(C(N(C2CN(C(C3(C)CCCCO3)=O)C2)C)=O)coc(S(C)(=O)=O)c1 96446,N1(C(c2c(OC)nsc2)=O)CCN(C(=O)CC(C)N(C)C)C(c2cccnc2)C1 96447,c1(C(=O)NCCC(C)NC(C(Br)=C(C)C)=O)cccc2cccc(C)c12 96448,c1(C(C(=O)NCC2CC(NC(CSCC(N)=O)=O)C2)=O)ccc(Cl)cc1Cl 96449,C1(CC(=O)NCCOC(C)=O)C=CC(NC(=O)C=Cc2ccsc2)C1 96450,c1(C(=O)NC)cc(OC)ccc1C(=O)NC1CCN(C(=O)C(C)C(C)C)C1 96451,C#Cc1cccc(C(=O)N(CC(N2CCN(C(C3(Cl)CC3)=O)CC2)=O)C)c1C 96452,c1(OC)nccnc1NC(c1csc(C(=O)N(CCO)Cc2ccccc2)n1)=O 96453,Cc1ccc(C)c(CC(=O)NC2CN(C(C34CC(CO)(C3)OC4C)=O)C2)c1 96454,C#CCC(C(=O)NCCOC1CCN(C(=O)CC(=O)NCC(F)(F)F)C1)C1CC1 96455,C1(CC)(NC(=O)CCCCN(C)C)CCN(C(=O)CSCCOC)CC1 96456,C1(COC)(CNC(=O)CC(C)SC)CCN(C(=O)C(C)CC(C)C)CC1 96457,CC1(C)CC(C(=O)NC2CCN(CCF)C2)CN1C(=O)CCC(=O)c1ccc[nH]1 96458,c1(NC(C2(OC)CCCN(C(=O)OC(C)(C)C)C2)=O)ccc2ccc(O)cc2c1O 96459,c1(OC)ccc(C(N2CCCC(CNC(=O)CCc3ccoc3)C2)=O)c(Br)c1 96460,c1(NC(C2(C)CCCN2C(c2cnc(O)[nH]2)=O)=O)ccn2ncnc2c1 96461,N1(C(c2c(C)cccn2)=O)CCCN(C(c2c(F)ccc(Cl)c2F)=O)C(C)C1 96462,c1(C(C)C)cnn(C)c1C(=O)NCC1(O)CC(NC(=O)CC2CCS(=O)(=O)C2)C1 96463,CC1(C)OC(=O)CC1C(N1CCC12CN(C(c1ccc(Br)cc1)=O)C2)=O 96464,C1(C(=O)OCC)CCN(C(C2CC(NCc3ccnnc3)C2)=O)CC1 96465,c1(CC)oc(C)cc1C(N1CC2CC2(CNC(c2sc(C)cc2OC)=O)C1)=O 96466,C1(NC(c2ccc(C(=O)O)o2)=O)CCCC1n1cc(Cn2cncn2)nn1 96467,C1(CNCC(COC(C)=O)C)C2CC3CC(C2)CC1C3 96468,c1(C(=O)NC2(C)CC(NC(c3ccc(CO)o3)=O)C2)cnc2scnc2c1 96469,CC(CC(F)F)C(=O)NCC(CO)NC(c1sccc1NS(C)(=O)=O)=O 96470,C(=O)(CCCCC(N)=O)NCC(S(C)(=O)=O)CNC(C1CC1C#N)=O 96471,Cc1cccc2ncc(C(N3CCC(C)CC3CNC(c3c[nH]c(=N)o3)=O)=O)n12 96472,C1(CNC(CC(=C)C)=O)CCC2(CO1)CC(NC(=O)C=CC1CCC1)C2 96473,N1(C(=O)OC(C)(C)C)CC(C(=O)Nc2ccc(Cc3cncs3)cc2)C2CC12 96474,CCCC(C)(CC)NC(C1(NC(=O)CNC(=O)CC(C)C)CCN(C)C1)=O 96475,C(C(F)(C(=O)NCC1CN(C(N)=O)C1)C(C)C)NC(C(CC)(C)C#N)=O 96476,C(=O)(C1CCCc2c[nH]nc21)NC1(CC=C)CN(C(=O)C(C)C(C)(C)C)C1 96477,Cn1nc(C(=O)NC2CC3(CCCN(c4nnnn4C)C3)C2)c2cc(F)ccc12 96478,C1(NC(=O)C=Cc2cnc[nH]2)CC2(C1)CC(C(=O)NCC1CCC(F)(F)C1)C2 96479,c1(C(=O)NCC(CNC(c2c(CC)nc(C)[nH]2)=O)F)cc(O)cc(F)c1 96480,c1(C(=O)NCCCN(C2CCN(C(C)C)C2=O)C2CCC(C)(C)O2)cnc(S)nc1 96481,N1(C(C2CCN(C(=O)COc3ccccc3)C2)=O)CC2COC(=O)C2C1 96482,N1(C(C2CC23CC(OCc2ccc(O)cc2)C3)=O)CCC(F)(F)C(O)C1 96483,N1(C(c2noc(CC)c2C)=O)Cc2occ(C(=O)NCCC3CC(F)(F)C3)c2C1 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96501,N1(C(c2c(Cl)cnc(C)n2)=O)CC2(CCC2)CC1CNC(=O)CCc1ccon1 96502,C1(NC(c2cnccn2)=O)CCC2(CC1)CN(C(c1ccoc1Cl)=O)CCO2 96503,c1(CNC(Cn2cc(C3(C)CC(OC)(OC)C3)nn2)=O)ccc2nsnc2c1 96504,n1(CC)nnc(C(N2CC(NC(=O)CC3CCCCC3F)C2)=O)c1C 96505,C1(SC)CN(C(=O)Cn2cnc(=N)[nH]2)CC1NC(C1(C)CCCO1)=O 96506,C12(CNC(C3N(C(C)C)CCC3)=O)CC1CN(C(c1cc(C3CC3)nn1C)=O)C2 96507,N1(CC2CCN(C(=O)COC3CCCCC3)C2)CC2C3C=CC(CC3)C2C1 96508,C#CCCCC(=O)NCCN(C(=O)CNC(=O)COCC=C)C(C)C 96509,C1(NC(c2n(C(C)(C)C)ncc2)=O)CCC2CC1CN2C(C1(C)CCOCC1)=O 96510,c1(C(N2C(CNC(C=CSC)=O)CC3(CCC3)C2)=O)cc(O)nc2cnccc12 96511,C(=O)(CC(O)C(Cl)(Cl)Cl)NCCC(C)(C)CNC(c1nc2ccccc2s1)=O 96512,C1(C(N(CCC)CCNC(=O)C(C)(C)C2CCOC2)=O)CCC(O)CN1C 96513,O=C1CN(C(=O)CCc2nc(O)n[nH]2)C(C(=O)NC2CCC3(CC3)C2)CN1 96514,C(=O)(C1CSc2ccccc21)NC1C(NC(c2cccc(S(C)=O)c2)=O)CCC1 96515,C1(C(=O)OC)(OC)CN(S(=O)(=O)CCc2ccsc2)C1 96516,c1(OC)ccc(F)c(C(=O)NC2CC2CNC(=O)CCOC(C)CC(C)C)c1Cl 96517,C1(C(=O)OC)CCC(CC(=O)NCCCNC(c2cccn2C)=O)CC1 96518,CC1(C(=O)NCCC2(O)CCN(C(=O)CC3CSC3)C2)CCC(F)(F)CC1 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96537,N1(C(c2n(CC)ncc2Cl)=O)CCC(C2CCN(C(=O)C(C)=C3CC3)C2)C1 96538,Cc1coc(C(C)C)c1C(=O)NCCCC1CN(C(=O)C(C)OC2CC2)CCO1 96539,N1(C(C2C(OC)CC2)=O)C2CCC1C(F)C(NC(=O)Cc1cnccn1)C2 96540,CC1C(=O)CCC(C(=O)NC2(CF)CCN(C(c3cscn3)=O)C2)C1(C)C 96541,c1(-c2ccc(C(=O)OC)c(F)c2)ccc2c(c1)OC(=O)CC2C 96542,CC1(C)C(NC(=O)C2=CCCC2)CCN1C(c1csc(Br)n1)=O 96543,Cc1ccc(C(=O)NCC(c2ccccc2)NC(=O)C(F)C2CCC2)c(F)c1F 96544,c1(COC(C2N(CC(=C)Cl)C(Cc3ccccc3O)C2)=O)ccc(SC)cc1 96545,C(c1cnc[nH]1)=CC(=O)NC(CN(C)C(C12CC(CO1)C2)=O)Cc1ccccc1 96546,C(C(C)C(=O)NC1CCC1NC(=O)C(C)(C)C)OCC 96547,N1(C(C2CN(C(N)=O)C2)=O)CC(O)(CNC(=O)COC2CCOC2)C1 96548,Cc1ccc(C)n1CC(=O)NC(C)CCNC(c1cccn1C1CCCC1)=O.C1(C)CC1 96549,c1(C(=O)NC(CC(C)C)CNC(C2CC2C#N)=O)c[nH]c2c(F)cccc12 96550,N1(C(CC=CCNC(=O)Cc2cccc(O)c2)=O)Cc2cccnc2C1 96551,N1(CC(F)F)CCn2nccc21.CC(CN(C)C)CC(=O)N1CC(CC(F)C=O)C1 96552,C#CCCCC(=O)NC1CCC(CCNC(c2ccc(Cl)cc2)=O)C1 96553,c1(OCC)cc(C(=O)N(C2CCN(C(=O)C=C(C)C)C2)CCO)ncn1 96554,C1(C(N2C(C)CCCC2)=O)CN(C(=O)Nc2c(O)ccc(F)c2F)CC(F)(F)C1 96555,C1(OC)CC(NC(=O)CN2CCP(C)(=O)CC2)CN(C(C2CSCCS2)=O)C1 96556,C(c1ccc(F)cc1F)=CC(=O)N(CC(CNC(c1c(C)cns1)=O)O)C 96557,CS(=O)(=O)C(CNC(=O)Cc1cc[nH]c1)CNC(C1(F)CCOC1)=O 96558,O=C(CCCOc1cccnc1)NCC1CN(CCO)C1.c1(CC)csc(C(Cl)Cl)n1 96559,c1(C(=O)NCC(CNC(c2c(C)ccn2C)=O)C)cccc2[nH]cc(Cl)c12 96560,CC1(C)CC(CC(=O)NCC(=C2CN(C(C3(C4CCC4)CC3)=O)C2)F)CO1 96561,Cc1cc(C(=O)NCCC2CCC(NC(c3ccc(Cl)c(F)c3)=O)C2)cc(O)n1 96562,N1(C(Cn2c(C)cnc2)=O)CCN(C(=O)CCCCC#N)CC1C 96563,C1(CNC(C2C(C)(C(C)C)C2)=O)C2CN(C(=O)CCc3c(N)cnn3C)CC12 96564,c1(C(=O)NCCCN(C(C2CC(C(C)C)OCC2)=O)C)c(F)cc(O)cc1F 96565,C(=O)(C(C)(C)CSC)NCCn1cc(C(=O)NC(CC)(C)CC)nc1 96566,N1(C(c2csnn2)C)CCC(C2(NC(=O)CCC(C)(C)C)CC2)CC1 96567,C1(C(N(CCCOCCNC(c2ccc(C)cc2)=O)C)=O)CCC2(CCC2)C1 96568,n1(CC)[nH]cc(C(=O)NCC2CC(NC(=O)C=CC(=O)OC(C)C)CCO2)c1=N 96569,C1(C(C2CC(C)CN2C(N2CCNCC2)=O)C)CN(C(=O)C2=C(Cl)CCC2)CCN1C 96570,C12(CNC(COCC)=O)CC1CN(C(=O)Cn1cc(I)cn1)C2 96571,Cn1cc(Br)c(CN2CCC(NC(=O)C(c3ccccc3)O)C2)n1 96572,C(=O)(C(C)CC(F)(F)F)N1CC(C)(C(=O)NCCCc2cc(C)no2)C(C)C1 96573,CC1(C)CC(C(N2CC3CCC3(CNC(=O)CSc3cn[nH]c3)C2)=O)C(C)(C)O1 96574,CCCC(C)CC(=O)NC(C)(C)CNC(C1SCCS1)=O 96575,N1(C(C(C(CC)CC)C)=O)CC(CNC(c2csc(C)n2)=O)OC2(CCC2)C1 96576,C1(C(=O)NC(C(C)C)CNC(C2(S(N)(=O)=O)CCC2)=O)CC2(CCCCC2)CO1 96577,n1(CC)cnc(C(N2CC(O)(CCNC(=O)C=CC3CC3)C2)=O)c1 96578,c1(-c2nc(Cc3cc(C)nc(C)n3)nn2C(C)CN(C)C)nc2nc(C)ccn2n1 96579,N1(C(CN(CCCCC)C)=O)CC(NC(=O)COCCCCC)CCC1C 96580,C1(CNC(CCC=CC)=O)CCCN(C(c2cn(C)nc2C(F)(F)F)=O)C1 96581,N1(C(c2cc(COC)sc2)=O)CC2CC1CN2C(=O)CC1CCOC1=O 96582,CC1CCc2[nH]c(C(=O)NCCNC(C3(CCO)CC3)=O)cc2C1 96583,C(C(=O)N(OC)C(C)CC)n1cc(CNC(c2cncc(C=C)c2)=O)nn1 96584,C1(NC(C2(CC#C)CC2)=O)(COC)CCN(C(c2ccc(CC)cc2O)=O)CC1 96585,c1(SC(c2cc(C)no2)C(=O)NCC(C)(C)OCC(=O)OC)ccccn1 96586,c1(OCC(=O)NCCCNC(C(C)(C)CF)=O)ccc(Cl)c2ccccc12 96587,C(=O)(C(C(C)C)c1cnc(C)s1)NC(CC(C)NC(C=C(C)Cl)=O)C 96588,Cc1c[nH]cc(C(=O)NCCC2(O)CCN(C(c3ccc(Cl)cc3N)=O)C2)c1=O 96589,c1(SC)c(C(=O)N(C)CCN(C(C2CC2C2CCC2)=O)C(C)C)cccc1F 96590,CC1(C)C(CO)CN1C(=O)C(C1(O)CCC1)NC(=O)C(O)CN1CCCC1 96591,CCCCC(C(=O)NC1CCN(C2CC2)C1=O)NC(=O)CC(=O)NC 96592,N1(C(CCCC(C)=O)=O)CCCC2(C1)C(NC(c1cccs1)=O)CCN2C 96593,CCCCN=C(NCc1cc(Br)ccc1Cl)N(C)Cc1cc(C)on1 96594,c1(C(=O)NC2CC(F)(CNC(c3cc(CC)nn3C)=O)C2)cc2ccccc2o1 96595,CC(C)CC(C)(CNC(C1CC(CF)C1)=O)NC(=O)CN1CCCCCC1 96596,C1(NC(CNS(C)(=O)=O)=O)CC(CNC(=O)CCc2cn[nH]c2)C1 96597,N1(C(c2cn(CCC)nc2)=O)CCN(C(=O)C2=CCCSC2)C(CC(C)(C)C)C1 96598,c1(C(=O)NC(CNc2nccc(OCC)n2)C2CC2)[nH]c2ccc(F)cc2c1C 96599,c1(NC(CC(=O)NCC2CC2CNC(C2(F)CCC2)=O)=O)ccccc1O 96600,C1(C(N2CC(CCOC)C2)=O)CCC2CCC1N2C(=O)CCc1cn(C)cn1 96601,C#CCC(CC#C)C(=O)NC(C)(CC)CCNC(c1ccc(Br)c(C)n1)=O 96602,C(CCC(=O)NC(C)(CNC(C1(c2ccccc2)CC1)=O)C1CC1)OCCOC 96603,CCCC(C)(C)C(=O)N1CC2CCCC2C1.c12ccccc1n1cc2nn1 96604,C(=O)(C(O)C(C(C)C)OC)N1C(C(=O)NC2CCN(C(CC)=O)C2)CC(F)(F)C1 96605,C(CO)(C(C)(C)CO)NC(C(C)CNC(=O)CCn1cccc1)=O 96606,N1(C(=O)CSc2nncs2)CCCC(NC(C2CC2(F)F)=O)CC1 96607,C1(C(=O)NCCCC(CCC)NC(=O)C(=O)NCC)COC2COCC2O1 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96625,CC1CC(NC(C2CC(F)(F)C2)=O)CCN1C(c1cc(CO)ccn1)=O 96626,N1(C(C2(SC)CC2)=O)CC2CN(C(C34C5CC(CC35)C4(F)F)=O)CC2C1CO 96627,N1(C(=O)NC2C(C)NCCC2)CCOC2(CCS(=O)(=O)C2)C1 96628,CCC(CC)CC(=O)NC1CCCCC1NC(=O)C(C1CCCC1)OC 96629,c1(C(N2C(CNC(CC=C)=O)CC2)=O)cn(CC(c2ccccc2)=O)nn1 96630,C1(C(=O)NCc2cc(C)sc2)(NC(C2CCCN(C)C2)=O)CCN(C)C1 96631,c1(C(N(CC(C)O)CC(C(=O)NC(C)C)=O)=O)cnc(-c2ccccc2)[nH]1 96632,C1(CCC=C)CCCCN1C(=S)Nc1ccc(S(C)(=O)=O)cc1 96633,c1(C(=O)NCCC(C)N(C(CC(CC)O)=O)C)[nH]nc2ncnc(O)c12 96634,N1(C(COCCOC)=O)CCCCC1CC(=O)NC(C)C1CC1 96635,N1(C(Cc2ncn(C)c2)=O)CC=C(C(=O)NCCC2CCCC3CC23)C1 96636,CC(CC(=O)N1CCCCC1C1(NC(=O)C(=Cc2c[nH]cn2)F)CC1)C(C)(C)C 96637,c1(N2CCC(C)C(F)(F)CC2)nc(=NCC2COCC2(C)C)[nH]c2c1CCCC2 96638,C(C(=O)N(C)Cc1ccncn1)(C(C)O)NC(c1c(CC)cco1)=O 96639,CC(C)CC(=O)NC(c1cn(C)nn1)C(=O)NC(C)CC(N)=O 96640,NC(=O)CC(O)C(=O)NCCC1(NC(=O)COC2CCCCC2)CCC1 96641,CC1CCn2ncc(C(N3CCC(C)C(NC(=O)C(F)C(C)(C)O)C3C)=O)c2C1 96642,C(=O)(C(F)(F)C1(O)CCC1)N(CCCCN(C(C(N1CC(C)C1)C)=O)C)C 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96660,Cc1[nH]cc(C(=O)NCC23CC2CN(C(c2ccnn2C(C)C)=O)C3)c(=O)c1Cl 96661,C12(C(N3CC4C(C(=O)OC)C4C3)=O)CC(CO1)N(C(c1cc(C)cs1)=O)C2 96662,Cc1ccc(C(C)(C)C(=O)NC2CC(Cc3ccc(Cl)cc3)C2)cn1 96663,CC1CCCCN1CC(=O)NC(CC1CCCC1)C(=O)N1CC(C)(C(F)(F)F)C1 96664,C(CN=c1nc(Cl)[nH]c(C)c1C#N)N(c1cc(C)ccc1F)C(=O)COC 96665,N1(C(c2c(C)cn(C)c2)=O)CCCCC12CC(NC(C1CCCCS1)=O)C2 96666,Cc1cn2cc(C(=O)NCC3CN(C(C4OCCC4C(C)C)=O)C3)sc2n1 96667,C(=O)(C(C)(C)CC(=O)NC1CCCC1(C)CN(C(=O)C(C(C)C)SC)C)OC 96668,CCC(CC)(CO)C(=O)NCCOCCCN(C)C(c1cn(C)ccc1=O)=O 96669,C1(NC(C2=C(C)CC2)=O)COC2(CCN(C(c3cccc4ccnn34)=O)C2)C1 96670,c1(CC(=O)NCCCN(C(c2cn(CCC(C)C)nn2)=O)CCO)ccccc1F 96671,N1(CC(=O)NC(C(=O)OCC)CC(C)C)CCCC(CC2CCCCCC2)C1C 96672,c1(C(=O)NC(CN(C(=O)CCC2CCCCO2)CC)C)cnc2[nH]nc(O)c2c1 96673,N1(C(C=C(CC)CC)=O)CC2CCCN(C(=O)CCc3c(C)nn(C)c3C)C2C1 96674,N1(C(C2(C=C)CCN(C(=O)CC(=O)OC)C2)=O)CCc2nc(O)[nH]c2C1 96675,C(=O)(C1=CCCOC1)N1C(CCNC(C2CC2(Cl)Cl)=O)CSCC1 96676,S(=O)(=O)(c1cccc(F)c1)NCC(=O)N(C)Cc1ccc(F)cn1 96677,c1(COC)nc(NCCS(=O)(=O)N(C)C)cc(N2CC3C(C2)C3(C)C)n1 96678,N1(C(CC2CC(C)(C)C2)=O)CCN(C(=O)C(O)C2CC2)C2COCC12 96679,Cc1cc(=NCC2(C)CC2(F)F)[nH]c(=NCCN2CCCC2)[nH]1 96680,c1(-c2cn(C3CCN(C(C4CCN(CC(C)C)C4)=O)C3)nn2)cc(F)ccc1F 96681,CN1CCC(C(=O)NC(C)(C)CN2CCN(C(C3(C)CC3(F)F)=O)CC2)C1=O 96682,C1(NC(Cc2ccc(OCC)cc2)=O)CC(C)CN(C(c2cscc2C#N)=O)C1 96683,N1(C(CCOCC#C)=O)CC2CCCC(N(C(=O)CN(C)C(=O)OC)C)C2C1 96684,N1(C(CCNC(=O)NC)=O)CCC(CNC(c2ccc(C(N)=O)cc2)=O)C(C)C1 96685,C1(C(=O)NCC2N(C(C(C)SC)=O)CC2)CCCN(C(=O)OC(C)(C)C)C1 96686,c1(CC(=O)NC(CC)CN(C(=O)CN(S(=O)(=O)CC)C)C)cccc2c1OCO2 96687,C(=O)(C1=CCCC1C)NC1CCC(C(=O)NCC2CC(C(=O)OC)C2)C1 96688,c1(C(N2CCC(CCNC(C=COCC)=O)CC2)=O)oc2c(c1C)C(=O)CCC2 96689,n1(CC)c(N2CCN(CC(=O)NC3CCOCC3)CC2)nnc1-c1ccoc1C 96690,C1(NC(CC2CCN(C(C)C)CC2)=O)CC2CN(C(=O)CS(N)(=O)=O)CC2C1 96691,c1(NC(C2(N(C(CSC(C)C)=O)C)CC2)=O)cnn(C2CCC2)c1 96692,c1(CN(C2(C(=O)OC)CCOC2)C(C)(C)C)cc(Br)ccc1OC 96693,C1(CNC(CC(C)C2CC2)=O)CCCCN(C(C2CCCC(O)C2)=O)C1 96694,N1(C(CCCN(C(C)C)C)=O)CC(C)(C)CC1CNC(c1[nH]nnc1C1CC1)=O 96695,N1(C(COCCNC(c2c(C#C)c[nH]n2)=O)=O)CC(C)CCC1CC 96696,N1(N2CCCC(C(=O)NCCNC(=O)C(C)C)C2)CCC(C)CC1.C(=O)OC 96697,c1(C(N2CCC3(NC(Cc4c(C)noc4C)=O)C(C2)C3)=O)ccc2nn[nH]c2n1 96698,c1(CC(=O)NC2CCCCC2NC(C2CC3C=CC2C3)=O)cccnc1Br 96699,C1(OC)CC2CC(C(=O)Nc3cccc(CNC(=O)C=CCF)c3)CC12 96700,c12n[nH]c3cc(ccc13)C(=O)NC2=O.c12nc[nH]c1NC2=O.N1(CC)CC(C)C1 96701,c1(-c2ccc(C(=O)NCCC3(OC)CN(C(C=NOC)=O)C3)s2)cccc(F)c1 96702,Cc1ccc2c(Nc3ccc(CCC(N4CCC(F)CC4)=O)[nH]3)ncnc2c1 96703,C(c1ccc(=N)[nH]c1)=CC(=O)NC1CC(N(C(Cc2ccn(C(C)C)n2)=O)C)C1 96704,CC1CN(C(=O)C(c2ccnn2C)O)CC1CNC(c1csc2cncn12)=O 96705,c1(-n2c(C(C)OCCC=C)nc(C3CCOCC3)n2)cccc2ccccc12 96706,c1(CNC(C(=O)NCc2cc(C(F)F)cc(F)c2)=O)cccc2c1OC(F)(F)O2 96707,n1(CCC)cc(C(=O)NCC2C=CC(NC(=O)C(C)SCC)C2)c(C)n1 96708,C12(CC(F)(F)C1)C(=O)N2.C1(CCNC(C2CC(CC)C2)=O)CCCC(C)C1 96709,CCCC(CCC)CC(=O)NC(C)(CO)C(=O)NCC(O)C1(Cl)CC1 96710,CP(C)(=O)CCC(=O)N1CCCCC(CCC(=O)NC2CC3C=CC2CC3)C1 96711,CCC(C)(F)C(=O)NCCN(C(=O)COCCOc1ccncc1)CCOC 96712,N1(C(CN(CCC)C)=O)CCC(CNC(=O)C(c2ccc(C)s2)C)C1 96713,c1(CCC(=O)NC2C(CNC(Cc3cc(C)sc3)=O)C2)cnc2ccccc2c1 96714,N1(C(CC2(C=C)CC2)=O)CCOCC(CNC(c2c(C(C)C)cccc2C)=O)C1 96715,C(=O)(C1CC(=O)Nc2ncn(C)c21)N1C(C)CN(C(C2CCSCC2)=O)CC1 96716,c1(N(C)C)cc(Cl)cc(CNC(=O)C(=O)NC2CCOC(C(F)(F)F)C2)n1 96717,C1(C(N2CC(CCNC(=O)C(C)N(C)C(C)=O)(OC)C2)=O)CCNC(=O)C1 96718,c1(SC)ncc(C(=O)NC2(C)CCN(C(=O)C=CC3CC3)C2)c(O)n1 96719,c1(CC)ccc(C(N2CCC(C(=O)NCC3CCC(F)(F)C3)C2)=O)cc1 96720,N1(C(CN(C(C)=O)C)=O)CCCCC(CNc2ncc(C)c(C)n2)C1 96721,C(=O)(C1OCCn2ccnc21)NCCCN(C(C(CC)(C)O)=O)C 96722,C=CCCC(C(=O)NC1CC(CO)(CO)C1)NC(c1ccc(C)nn1)=O 96723,c1(C(C(=O)NCC)N(c2cnn(C(C)C)c2)CC2CC2)cc2cc(Cl)ccc2s1 96724,CS(=O)(=O)c1cc(C(N2CCN(C(=O)C=CC3CCCO3)C(CCO)C2)=O)cs1 96725,c1(C(=O)NCC2(CCCNC(C=COC)=O)CCCC2)ccc(P(C)(C)=O)nc1 96726,N1(C(CCC(C)=O)=O)CC2CC(C1)N(C(c1cccc(C3CC3)c1)=O)C2 96727,c1(C(N2CC(C)C(NC(c3ccc(CC4CC4)s3)=O)C2)=O)coc2c1CSC2 96728,N1(CC)CCCCC1C(=O)OC(C)C(=O)NCCNC(=O)N(C)C 96729,C=CC(C)(CC)C(=O)N1CCC(N(CCO)C(c2ccc(=O)oc2)=O)CC1 96730,c1(CC)nc[nH]c(=NCC(C)(C)NC(=O)CC2CCC(C)(C)CO2)c1F 96731,c1(N2CC=CC(NC(COC(CC)(C)C)=O)C2)cc(C)ncc1C#N 96732,C12(C(N3CC(C=C)(O)C3)=O)CCCC1CN(C(=O)CS(=O)(=O)CCOC)C2 96733,c1(C(N2CC(NC(CC=CCC)=O)CC2(C)C)=O)cnn2c1CC(C)CC2 96734,C#CCCCC(=O)NC1(CCNC(c2cc(C(F)(F)F)n[nH]2)=O)CC1 96735,CCC(C(=O)N(C(C)CCNC(c1cn(C)cn1)=O)C)NC(C)=O 96736,C1(CNC(C2(CC)CCCC2)=O)CCN(C(C23CCC(CC2O)C3)=O)CC1(F)F 96737,c1(OC)cc(C(=O)NC2CN(C(C3CCC4CC34)=O)CC2OC)ccc1C 96738,c1(C(=O)NC2C(NC(C(C)O)=O)C2)cc2ncccc2[nH]1 96739,C(=O)(C(CSC)c1ccccc1)NCCN(C(=O)C(C)(C)N(C)C)CCC 96740,C(=O)(CC1OCc2ccccc21)NCC(CNC(CCC=CC)=O)(C)O 96741,C1(C(=O)NCC2(C)CCN(C(C)=O)C2)CC2(CCOCC2)CN1 96742,N1(C(=O)C=C2CCOCC2)CCC2CN(C(C3(C4CCCO4)CC3)=O)CC2C1 96743,CC(C)CCCCC(=O)N1CCN(C(=O)CCCC(=O)c2ccccc2)C2CC12 96744,C(=O)(C1CCc2nnc(C)n21)NCc1scc(CNC(C(CC=C)(C)C)=O)n1 96745,C1(C(=O)OC)(C(=O)NCCCC(=O)NCCC2CCCCO2)C=CCC1 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96763,c1(C(N(CC(CNC(CC2C(CC)C2)=O)(C)C)CC)=O)cc(=O)cc[nH]1 96764,c1(OC)cccc(C(=O)NC(c2ccccc2)C(=O)NCCC(O)C(C)C)n1 96765,Cc1noc(C(=O)N(CCC(C)NC(=O)C(C)Cc2c(C)noc2C)C)c1C 96766,c1(OC(C)C(=O)N(C)CC2(O)CN(C(C3COCCO3)=O)C2)cccnc1 96767,N1(C(C=NOC)=O)CCOC(COC2CCN(C(c3nnc(S)n3C)=O)C2)C1.N 96768,C12(C(N3CC(Cn4cc(C(CC)O)nn4)OCC3)=O)CCCCC(=O)N1CCC2 96769,c1(OC)cc(C(=O)O)ccc1CNc1ccc(-c2nncs2)cc1 96770,C1(CC(=O)NC(C(=O)NCc2cc[nH]n2)C2CCCC2)CCC(O)C1 96771,C1(COC)(CNC(c2sccc2Cl)c2nnnn2Cc2ccccc2)CCCO1 96772,C1(n2cc(C3C(c4nc(C)[nH]n4)CCO3)nn2)CCCN(C(C2CC2C)=O)C1 96773,c1(CN(CCN(C(c2csnc2C)C(=O)NCCSC)CCC)C)ccccc1Br 96774,CCCCCC(C)(CC)C(=O)N1CC2(CCC2NC(=O)CSC(F)(F)F)C1 96775,n1(CC(=O)NC2(C)CN(C(C(CC)O)=O)C2)[nH]cc2c(=O)ncnc1-2 96776,N1(C(CC)C(=O)NCCC(C)NC(=O)Cn2nnc(=N)[nH]2)CCN(CCO)CC1 96777,C1(C(=O)Nc2c(SCC)cc(F)cc2)CCn2c(O)nnc2C1 96778,c1(CC)cccc(NC(c2ccc(OC3CCCC3)nc2)C)c1 96779,Cc1cc([N+](=O)[O-])c(S(=O)(=O)N2CCC(C(=O)N(CC(=O)O)C)C2)cc1F 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96798,c1(CNC(N(CCOCCO)CC)=O)cccnc1S(C)(=O)=O 96799,C(=O)(CC(C)(C)C(=O)N1CC(C(=O)NCC2(O)CN(C)C2)C(CC)C1)OCC 96800,C1(CNC(COCCC=C)=O)CCC(C)(C)CN1C(C1CCCCS1)=O 96801,CCCCN=C(NCCCc1cc2ccccc2[nH]1)NCC1CC(O)C1(C)C 96802,C1(c2cn(CCOC)nn2)CCCN(C(C2CC3(CO)CC2C3)=O)CC1 96803,C(C)(C)(CCC(=O)N1CCCC(C(N2CCC(C)(C(N)=O)C2)=O)C1)OC 96804,N1(C(c2c(C#C)c[nH]n2)=O)CCC(F)CC1C(N1CCC(C)CC1)=O 96805,C(=O)(C(C)CC(F)(F)F)NC1(CC=C)CN(C(=O)C(COCC)N=[N+]=[N-])C1 96806,C=C(C)CCCC(=O)NCC(CCOC)NC(c1coc(C(C)OC)n1)=O 96807,CC1CN(CC(C)(C)O)CCN1C(=O)NCC1(C)CC=CCO1 96808,C(=O)(CC(C)CC(F)(F)F)NCC1N(C(c2cnc(SC)s2)=O)CC(O)C1O 96809,N1(C(C2C(CC)OCC2)=O)CC(C)(C)CCC1CNC(c1cc(C)nc(O)n1)=O 96810,C1(C)(C(N2CC(C)(NC(=O)CN3CCSCC3)C2)=O)C2Cc3ccccc3C12 96811,N1(C(C2(C#C)CCC2)=O)CCC(NC(c2ccccc2)=O)C(CC2(SC)CC2)C1 96812,N1(C(c2cccc(C)c2C)=O)CC2CCC1(CNC(c1[nH]c(O)nc1C)=O)CC2 96813,c1(CC(N2CC(NC(CCOC)=O)C(C(F)F)C2)=O)ccc(OC(F)F)c(F)c1 96814,CC1(C)C2CC(NC3(C)CN(C(=O)CNS(=O)(=O)C4CC4)C3)CC12 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96832,CCC1=NOC(CC(=O)NC23CC2CN(C(=O)COc2cccnc2)C3)C1 96833,Cc1cc(CNC2CCN(C3CCN(C(C4(C(N)=O)CC4)=O)CC3)CC2)ncn1 96834,CC1(C(N2CCN(C3CCCN(C(C4(C(N)=O)CC4)=O)C3)CC2)=O)CCNC1=O 96835,c1(C(=O)NCC(C2CCOC2)NC(c2n(C(C)C)nnc2)=O)cnc2n1CCC2 96836,N1(C(COc2ccc(C(C)=O)cc2)=O)CC(C2(NC(=O)CC#N)CC2)C1 96837,C1(NC(Cc2c(C)cccc2)=O)CCN(C)C12CCCN(C(=O)C(F)C(C)C)C2 96838,c1(C(=O)NC2CC(CNC(c3c(CC)n(CC)nn3)=O)C2)cnc(O)n(C)c1=O 96839,C1(C)(NC(c2n(C(C)C)nnn2)C(C2CCOCC2)C)CCC(=O)N(C)C1 96840,CC1(C(=O)NCc2ccoc2C(=O)NC2CC(O)C2)CCC2CC2C1 96841,c1(SCC(=O)NCC2(NC(c3cc(Cl)ns3)=O)CC(F)(F)C2)ccc(O)cc1 96842,c1(C(=O)NCC(C)(C)NC(C23CCCCC2C3)=O)cc2c(cc1Cl)NC(=O)C2 96843,O(NC(=O)N(CCc1nn[nH]n1)C1CC1)CC(=O)OCC(=O)NC(C)C 96844,C1(C(=O)NC2C(NC(CC(C(C)C)O)=O)CC2)CC12C1CC3CC(C1)CC2C3 96845,C(=O)(C(C)(O)CCN(C)C)NCC(CCC)NC(c1cccc(C(F)F)c1)=O 96846,c1(NC(c2ccc(CC)o2)=O)cccc(C)c1C 96847,N1(C(Cc2c(C)noc2C)=O)C2CCC1(CNC(c1ccco1)=O)CC2 96848,c1(C(N2C(CNC(CC(=O)NCC)=O)CC(OC)C2)=O)cc2c(=O)[nH]ccn2n1 96849,c1(C(C(=O)N(CCNC(C(C)CO)=O)C)C)nc(F)ccc1Cl 96850,C1(C(=O)NCCCOC=C)C2CCCC2CN1C(=O)CN1CCCCC1=O 96851,N1(CC(=O)NC(C2CCCC2)CNC(C=CCOC)=O)CCC(C)C1 96852,c1(NC(C2C3CC(N)C(C3)C2)=O)c(Br)cc(Br)c2cccnc12 96853,Cc1cc(C(F)(F)F)nn1CC(=O)NC1CCCCC1N(C)C(c1ccc[nH]1)=O 96854,N1(C(CCCOCC)=O)CC2(CCN(C(=O)C(C)CCO)CC2)C1C(C)C 96855,CC1=C(C(=O)N2CC(NC(c3ccsc3CN)=O)C(C)C2)CCO1 96856,CCC(C(=O)NC1CC(C)(CNC(=O)C=CCOC(C)(C)C)C1)SC 96857,N1(C(C=C(CC)C)=O)CCC2(CCCN2C(c2cnc(C(C)(C)C)nc2C)=O)C1 96858,c1(C(COC)NC(=O)NC2CC23CC(O)C3)ccc(Br)cc1Br 96859,N1(C(CC(CCC)C)=O)CC(CNC(c2ccnnc2C)=O)OC(C)(C)C1 96860,Cc1ccc(C(N2CC(C(F)C(=O)N=c3ccn(CCF)[nH]3)C2)=O)c2c1CCCC2 96861,c1(CC(=O)NCCC2(NC(=O)Cc3ccncc3Cl)CC2)ccc(Cl)cn1 96862,CC(C)C(CCN(C(=O)CC1CCSC1)C)NC(=O)CC1CCC(=O)N1 96863,Cc1cc(=NCC2CCSC2(C)C)[nH]cc1S(=O)(=O)N1CCOC(CCO)C1 96864,Cc1c(NC(=O)N(C)CC2CCN(CC(F)F)CC2)cnn1C1CC1 96865,c1(CC(=O)NCCCN(C(C23CCCCC2C3)=O)CC)ccc(S(C)(=O)=O)cc1 96866,CC1CCC(CCC(N2CCC(Cc3cn(CC(=O)NC(C)(C)C)nn3)C2)=O)OC1 96867,Cc1nn(C)c2nc(C(=O)NC3CN(C(=O)COC4CCOC4)C3)cc(O)c12 96868,C1(C(=O)NC2C(O)C3CCCC23)CCN(C(=O)CCC2CC2)O1 96869,CCC(CCC(=O)NC(CC(=O)NC)C1CC1)NC(=O)C(C)(C)n1cnnn1 96870,C12(C(N(CCNC(c3c(CC)nns3)=O)CC3CC3)=O)CC3CC(C(=O)N1)C2C3 96871,N1(C(C=C2CCC(C)(C)CC2)=O)CCC2(CCC(NC(C3CCCO3)=O)CC2)C1 96872,CCCCCC(CC)C(=O)NC(C)C(C)(C)NC(c1ccc(CC)[nH]1)=O 96873,c1(CCC(=O)NC(C2N(C(c3cnc(SC)s3)=O)CCC2)C)ccnc(Cl)c1 96874,N12CCC(O)C(O)C1C2.c1(CC=C)ccc(OCC(=O)OC)c(OC)c1 96875,N1(C(C(C)=CC)=O)CC(NC(=O)CC2COCCO2)CC2(CCC2)C1 96876,N1(C(C=C(CC)CC)=O)CCN(C(c2cnn(C)c2COC)=O)C(C)C1C 96877,c1(NC(c2n(CCCF)nnn2)c2ncoc2C2CC2)cc(F)cc(F)c1 96878,N1(C(c2ccc(C3CC(=O)NC3)cc2)=O)CCC(F)(CNC(=O)C2=CCC2)CC1 96879,c1(C(C)=O)ccc(NC(=O)C(=O)NCC(Cc2ccc(Cl)cc2)C(=O)O)cc1 96880,Cc1ccc(CC(=O)NC2C=CCN(C(C3(CF)CC(F)(F)C3)=O)C2)cn1 96881,C1(NC(c2c(Cl)cn(CC)n2)=O)(CC)CCN(C(=O)CN2CCOCC2)CC1 96882,C1(NC(C(C)C#N)=O)CCOC12CCN(C(=O)CC1(C)CCS(=O)(=O)N1)CC2 96883,C(=O)(CCC(CC)NC(=O)C1=C(Cl)CC1)N1CC(O)(CC=C)C1 96884,c1(OC)ccc(CCCC(=O)N2CC(CCNC(=O)C(O)C3CC3)C2)cc1OC 96885,c1(OC(C)C(F)(F)F)ccccc1-n1cc(C2CCCC2O)nn1 96886,C(N=c1[nH]c(NC)ncc1Cl)N1CCC(Oc2c(OCC)ccc(C(N)=O)c2)C1 96887,c1(C2CC3(CC(CN(C)Cc4c(OC)c(Br)ccc4)C3)C2)c(F)ccc(F)c1Cl 96888,C1(C)(C(=O)NC(c2nn[nH]n2)CC)CC(NC(=O)CC(C)=C(C)C)C1 96889,c1(C(=O)NCC=Cc2c(OC)cc(Br)cc2)c(Cl)ccc2c1OCO2 96890,N1(C(CCSC)=O)CC(NC(c2cc(-c3ccncc3)no2)=O)CC12CCOC2 96891,C1(NC(C2CCC(C)(C)O2)=O)CC2CN(C(c3cc(O)ncn3)=O)CC2C1 96892,c1(CC)cc2c(N3CCC(CF)(NC(c4cnsc4C)=O)C3)nc(C)nc2s1 96893,c1(OC)nsc(C(C(=O)Nc2ccccc2)N(C2CCCC2)C)c1Cl 96894,c1(OC)cc(C(N2CC(C(O)C(=O)NCCC(=O)NO)C2)=O)n(C)n1 96895,c1(C(N2CCN(C(Cc3cncc(OC)c3)=O)C3C2C3)=O)cncc2sccc12 96896,C(=O)(C1CCCc2ncnn21)N1C2CC(CNC(C(C)N(CC)CC)=O)(OC2)C1 96897,C1(N2CCC(N(C(C(CC)C)=O)C)C2)CCN(CC)CC1 96898,C(CO)(CC(F)(F)F)NC(CCCN(C(c1n(CC)nc(C)c1)=O)C)=O 96899,C(=O)(C1CCOc2ccccc21)N(CCCN(C(C(CC(C)C)=O)=O)C)C 96900,c1(C(=O)NCC(CC)NC(c2ccccc2S(C)=O)=O)cccc(C#CCO)c1 96901,CC1(C)OC2(C(=O)NCC(C3CCCC3)NC(=O)CC3CCOCC3)CCC1C2 96902,N1(C(C(C)(C)CO)=O)CC2(CCC2NC(=O)Cc2cc(C3CC3)nn2C)C1 96903,S(=O)(=O)(C1CN(C(=O)OC(C)(C)C)C1)NC(C)CC1CCC(C)(C)CC1 96904,N#Cc1[nH]c(=NCC(C2CCCCC2)NC(C2(O)CCSCC2)=O)sc1Cl 96905,c1(N(C)CCOc2ccccn2)ccncc1S(=O)(=O)NCC1CC1(F)F 96906,C1(CNC(c2c(C)cnn2C)=O)CN(C(c2nccnc2Cl)=O)CCC1C 96907,C1(NC(C2CCC(=C)CC2)=O)CCCN(C(=O)CCn2cnc(C)cc2=O)C1C 96908,c1(C(N(CC(C)NC(COCCCC)=O)C(C)C)=O)cnc(SCC)s1 96909,N1(C(CCC(CC)C)=O)CC2CC(C1)CN(C(=O)CCC1CNC(=O)N1)C2 96910,CC(C)C(C(=O)NC1CC(NC(=O)C(C)N(C)C)C1)N1CCCCC1 96911,C(CCN=C(NCC(N1CCCC1)=O)N1CCc2sc(Cl)cc2C1)OC(F)(F)F 96912,C=C1CCN(C(=O)C(c2ccccc2)NC(c2cccn2C)=O)C1 96913,O=C(C#CC1CCOC1)NC1CCOCC1NC(=O)Cc1nc2ncccn2n1 96914,c1(C(N2CCCC(C(C)NC(=O)CSc3ccncc3)C2)=O)cnc(Cl)cc1Cl 96915,c1(NC(C2C3CN(C(=O)C(O)c4ccsc4)CC23)=O)cc(C(F)(F)F)ncn1 96916,c1(C(=O)NCC2(NC(c3ccc(F)s3)=O)CC2)cccc2cccnc12 96917,Cc1cnnc(O)c1C(=O)NC1CC(C(=O)NCCC(C)(O)C2CC2)CC1O 96918,C1(O)(CC#C)CC(C(=O)NC(C2CCN(C(=O)CC=C=C)C2)C)C1 96919,CC1CCN(C(=O)CCc2ccc(Cl)cc2F)CC1CNC(=O)CN(C)C(N)=O 96920,C1(CC(=O)NCC(c2ccccc2)O)CCN(Cc2ccccc2Br)CC1 96921,C(=O)(C(F)(F)CCn1cccn1)NC(CC(C)C)CNC(=O)CC12CC(C1)C2 96922,C(CC(C)(C)CC(=O)N1CC(c2cc(O)no2)C1)OC.C12CC=CCC1C(=O)NOC2=O 96923,C(N=c1[nH]c(=N)[nH]c(=NC2CCCCC2C(N)=O)[nH]1)c1cnc(C)o1 96924,CC(CC(=O)N1CC(O)(CCNC(=O)CCCn2cccc2)C1)CC(F)(F)F 96925,CC1OCCCC1C(=O)NC(C)(C)C=CC(=O)NC1(C2CC2)CC1 96926,c1(C(=O)NC2CC(CCNC(C=CC(C)C)=O)C2)cc2c(s1)CCS(=O)(=O)C2 96927,C(COCC(N1CC(NC(N)=O)C1)=O)(C(=O)N1CC(O)(C(F)(F)F)C1)N(C)C 96928,C1(C(=O)NC(c2nncs2)C)CN(C(C2CC2Cl)=O)CC12CCC2 96929,c1(CCCN(C(C2CCCN(CCCOC)C2)=O)C(C)C)nnc2ccccn12 96930,c1(C(CC)C)ccc(C(C(=O)NCCC2(C)CC2)N(C2CCCCCC2)C)cc1 96931,N1(C(C(C)(C)OCC)=O)CCC(N(C(c2sccc2F)=O)CC)CC1 96932,Cc1cc([N+](=O)[O-])c(Cl)cc1NC(c1ccc(NCc2ccn(C)n2)cn1)=O 96933,C1(CC(N2CCCC2Cc2ccccn2)=O)CCc2ccccc2N1 96934,c1(C(=O)NC2CCN(C(C(CCC)(C)O)=O)CC2(C)C)cccc2c1CC(=O)N2 96935,C1(CNC(c2ccc(Cl)cc2)=O)COCCN1C(c1cc[n+]([O-])cc1)=O 96936,Cc1ccc(O)c(C(=O)N(C)CC2CC(F)CN2C(C2CN3CCC2CC3)=O)c1 96937,N1(C(c2n(CC)ncn2)=O)C2CCC1CC(N(C(=O)CN1CCCCCC1)C)C2 96938,C1(CC)CN(c2nnc(CN(C)S(N)(=O)=O)n2C)CC(C)O1 96939,C1(NC(CCC(=C)C)=O)CCN(C(c2coc(C(F)F)n2)=O)CCC1CO 96940,c1(C(=O)NCCN(C(C(C)=C2CCC2)=O)C(C)C)cccc2c(C)ccnc12 96941,C(CC(=O)NCC1CN(c2cc(C(N)=O)nc(Cl)n2)CCCO1)(C(F)(F)F)OC 96942,C(=O)(C1=Cc2ccccc2C1)N(CC(C)NC(CC(C)c1ccccc1)=O)C 96943,N1(C(C(CN(C)C)O)=O)CCC2C(C1)CN2C(c1cnn2cccnc12)=O 96944,C1(NC(CC2CC(CC)C2)=O)CCC(CC(=O)NC(C)(C)CCN(C)C)CC1 96945,C=CC(CCC)CC(=O)NC1(CO)CCN(C(=O)Cc2csc(C)n2)C1 96946,c1(C(=O)NC2CN(C(=O)Cc3ccccc3F)CC2F)c(F)cc(F)cc1F 96947,N1(C(=O)CCc2nc(O)n[nH]2)CCC2CCN(C(C3CCCC(F)C3)=O)C2C1 96948,N1(C(c2n(CCOC)ncc2)=O)CC2CCCC2(NC(c2ccnnc2)=O)C1 96949,O=C(C1=CCCC1)NCCc1ccc(Oc2cccnc2)cc1 96950,C1(CC)CN(C(C2CC2[N+](=O)[O-])=O)CCN1C(=O)C#CC1(C)CC1 96951,CCCS(=O)(=O)CC(=O)NCC1(CCNC(c2cncc(NCC)c2)=O)CC1 96952,N1(C(c2ccc(C)nn2)=O)CCC2CCN(C(=O)C(C)CCO)CC2C1 96953,C1(C(C)C)CN(C(=O)C(C(C)C)OC(N)=O)CCN1C(c1cccc(Cl)c1)=O 96954,c1(CSCC)cc(C(=O)NCCCCCNC(C2CCC(C(N)=O)C2)=O)no1 96955,Cc1ccnc(C(O)CNC(C2CCCN2C(=O)OC(C)(C)C)(C)C)c1 96956,N1(C(C(COC)O)=O)CCCC(NC(=O)C(O)CCc2ccccc2)C1C 96957,Cc1cc(Br)cc2c1C(NCCC=Cc1ccc(Br)cc1)CC2 96958,C1(C(N2CC(=C(CNC(=O)Cc3ncc(Cl)s3)F)C2)=O)C2CCCCCCC12 96959,c1(C(N(C2CCCN(C(C3CC4(CCC4)CO3)=O)C2)CC)=O)cc2sccc2s1 96960,O=C1CSc2cc(C(N3CC4CCNCC(C4)C3)=O)ccc2N1 96961,Cc1cccc([N+](=O)[O-])c1NC(C1C=CC(C(=O)N=c2cc(CCO)[nH][nH]2)C1)=O 96962,CCC(C)C(O)CC(=O)NC(C(=O)NC1CCCC1(C)N(C)C)C1CCOC1 96963,C1(C(=O)NC(C2CCCC2)CNC(=O)COC2CC2)Cc2ccncc2N1 96964,N1(C(C=CC)=O)CC2CCC(C1)N2C(=O)NCCCCCl 96965,N1(c2nc(C)cc(N3CCC(CCOC)C3)n2)Cc2c([nH][nH]c2=N)C(C)C1 96966,Cc1c(CNC23CCC(C(=O)NCc4cccnc4)(CC2)C3)ccnc1Cl 96967,C(C)(C)(C(C)CC(=O)N1CC(O)(CO)C1)NC(CCC#CC)=O 96968,C1(C(N)=O)CC(F)CN1C(=O)CC1CCCC(NC(c2cnn[nH]2)=O)C1 96969,c1(CCN(C)C)nc(-c2cnc(CCC(=O)NC(C)(C)C)[nH]2)n(CCF)n1 96970,C1(OCC)CC2(C1)CC2C(=O)N(C(C)CN(C(=O)CCc1cccn1C)C)C 96971,c1(C(=O)Nc2cccc(CNC(c3cscn3)=O)c2)ncc2ccccn12 96972,CCC(C)C(O)C(C)C(=O)N(C(C)(C)CC(=O)NCC(Cl)C(C)(F)F)C 96973,C(=O)(C(F)CC(C)(C)NC(=O)CC(C)Oc1ccccc1)NCC1CN(CC)C1 96974,Cc1ccc(O)c(C(=O)NCC2CC(NC(=O)CC(C)C)C23CCC3)c1 96975,C(=O)(CC(F)(F)CC(F)(F)F)OCC.c12ccc(cc1)n(C)c2=O 96976,c1(C(CC(=O)NCC2(C)CN(Cc3cnc(C(C)C)[nH]3)C2)O)ccc(F)cc1 96977,N1(C(c2n(C)ncn2)=O)CC(NC(=O)Cc2ccc(Br)cc2Cl)CC(F)(F)C1 96978,C1(CCC(=O)NC2(C)CC(NC(c3ocnc3C(F)(F)F)=O)C2)NC(=O)NC1=O 96979,C=CC(C)CC(=O)NCC1(F)CCN(C(c2cc(C(F)(F)F)cs2)=O)C1 96980,C1(NC(CC(C)C)=O)(CO)CCCN(C(c2cn(Cc3cccs3)nn2)=O)C1 96981,C#CCC(CC(F)F)C(=O)NC1CN(C(c2nn(C)cc2C)=O)CC12CC2 96982,N1(C(C=CC(C)NC(c2ccc(SC)s2)=O)=O)CCCC1(C)CO 96983,c1(C(=O)NCC2(C(F)F)CCN(C(C(C)(C)C(N)=O)=O)C2)ccc2ccsc2c1 96984,CC(C)(C)CCC(F)C(=O)N1CC(C)(OCC(N2CC3(CNC(=O)OC3)C2)=O)C1 96985,C=CC(CCC)CC(=O)N(CC(CC)NC(c1sccc1OC)=O)C 96986,C1(NC(c2ccc(C(F)F)nc2)=O)CCCC(CNC(C2CCCC23CC3)=O)C1 96987,CC1CCN(C(=O)C(F)(F)F)CC1C(=O)Oc1c(C(=O)OC(C)(C)C)cccc1 96988,c1(C(=O)NCCCC(C)NC(C2CCC(=O)N2)=O)ccnc(C(F)(F)F)c1F 96989,CCCCCC(O)C(=O)N1CCCC(C(C)C(=O)NOCC(=O)OCC)C1 96990,C1(NC(C2C(=C)CC2)=O)CC(C)(NC(c2ccsc2OC)=O)C1 96991,N1(C(CCSCC(C)C)=O)CC(CNC(=O)CCNC(=O)NC2CC2)C2CC12 96992,C12(C(NOCC)=O)CCN(C(=O)CCc3ccccn3)CCC1C2 96993,c1(C(C(=O)NC(C(C)NC(C2(C(=O)N(C)C)CC2)=O)C)C)cccc(C#N)c1 96994,C12CC3OCCC3N(C1)C2.C1(c2ncn(C)c2)CN(C(=O)NC(C)(C)C)CCO1 96995,c1(C(N2CCCC(C(N3CCCC34CC4)=O)C2)=O)cccc2c(O)ncnc12 96996,C=C(C)CC(C(=O)NCc1cncc(C(=O)NCC2CC2Cl)c1)OC 96997,C(=O)(C(C)(C)CCCNC(c1coc(N(C)C)n1)=O)NC(CCC)(C)CO 96998,c1(CNC(CCOCC)=O)ccc2c(c1)CCN(C(c1c[nH]c(=NC)o1)=O)C2 96999,O=C1CCCc2ccc(CNC(N3CC4(CCSCC4)C3CCO)=O)cc2N1 97000,c1(C(=O)NCC2C(NC(c3cnn(C4CC4)c3)=O)C2)nscc1Br 97001,C1(C(N(C(CSC)C)C)=O)C2CCN(C(=O)C3=CCOCC3)CC12 97002,S(=O)(=O)(c1ccc(NCc2nc(Cl)cs2)cc1Br)NC(CC)C1CCC1 97003,Cc1[nH]nc(C(=O)NCC(O)CN(C)C(C2(C)CCCCC2)=O)c1C 97004,c1(-n2ccc(C(=O)NCCNC(C(C)C)=O)n2)ccc(F)cc1F 97005,Cn1cnnc1C(CO)NC(=O)CC1(NC(=O)CN2CCOC2=O)CC1 97006,c1(OCC)ccc(C(F)(F)F)cc1NC(=O)NC1CCCC(SC)C1 97007,C(CN=c1nc(COC)[nH]s1)C1N(C(CC2CC(OC)C2(C)C)=O)CCCC1C 97008,c1(COC)cc(C(=O)NC(C)(C)CNC(c2nnc(-c3ccon3)s2)=O)no1 97009,S(=O)(=O)(c1cccs1)NCC(N1CC2C(NC(c3c(CC)nn(C)c3)=O)C2C1)=O 97010,c1(CNC(=O)CC2CC(F)C2)n[nH]cc1C(=O)NCC#CC1CC1 97011,C(C(C(=O)NC(c1ccoc1)C)NC(=O)C(C)c1cc[nH]n1)OCC 97012,c1(C(=O)NCCC2N(C(C(C)C(F)F)=O)CCC2)csc2ccc(F)cc12 97013,N1(C(c2c(CC)noc2)=O)CC(C2CCN(C(c3ccnn3C3CC3)=O)CC2)C1 97014,N1(C(CCSC)=O)CCC(OCCNC(C2CC(C)(F)C2)=O)C1 97015,Cn1cnnc1SCC(=O)NCC1(F)CC(NC(C2(C(F)(F)F)CC2)=O)C1 97016,C(=O)(C(=O)N=S(C)(C)=O)N(CCC(C(C)C)NC(=O)C(=O)C(F)(F)F)C 97017,C1(C)(C(N(CC(C)O)CCNC(C2(CCCC)CCC2)=O)=O)CCOC1 97018,N1(C(C(CC)N(C)C(c2ccc(O)cc2)=O)=O)CC2(CCC(=O)O2)C1 97019,c1(OC)ncccc1C(=O)NC(C)CNC(c1[nH]c(C2CC2)nc1C)=O 97020,CCC(C)C(C(=O)N(CCC(=O)NCC(C)(C)O)CCO)N(C)C 97021,C1(C(N(C2CCCCC2NC(C2CCOCC2)=O)C)=O)CCCN(C2COC2)C1 97022,Nc1cccc(C(=O)NCCC2CCC(NC(=O)CC(C3CC3)C3CC3)C2)c1F 97023,n1(CC=C)cccc1C(=O)NC1CC(N(C)C(c2ccc(C(F)(F)F)s2)=O)C1 97024,N1(C(C(C(C)C)NC=O)=O)CCCCC(CNC(=O)CCC2CCN(C)CC2)C1 97025,c1(C(C(=O)NC(c2cn(-c3cccc(F)c3)nn2)C)(F)F)cccc(F)c1F 97026,c1(C(=O)NCC(c2cccs2)C)cc(CCNC(=O)CC2CCCC2O)on1 97027,Cc1ccc(=O)n(CC(=O)NC2CC(C)(NC(C3CCCC3CF)=O)C2)n1 97028,c1(C(=O)NC2CN(C(CC(C(C)C)O)=O)C(CO)C2)cc2ccccc2o1 97029,C=CCC(CC=C)C(=O)N1CCN(C(=O)CC2CC(=O)NC(=O)C2)CC1CF 97030,Cc1cc(Br)cnc1Nc1cncnc1NCC1CC(C(=O)OC(C)(C)C)C1 97031,C1(CNC(C(C2CC2)OC)=O)CN(C(=O)C(C(C)C)NC(=O)CC(C)C)CC1C 97032,C1(C)(SCc2nc(C34CC(C)(C3)OC43CCC3)on2)CCc2ccccc2O1 97033,CC(C#N)CCC(=O)N1CCC(CNC(=O)CCC2CCCCC2)CC1 97034,C(=O)(C1=CCCCC1)N(C)CC1CN(C(CC2(OCC)CCC2)=O)C1 97035,C(=O)(C(CC)C(F)(F)F)NC(CC(=C)Cl)C(=O)N1CC(C)C(O)C1 97036,N1(C(CC(CCC)NC(c2sccc2F)=O)=O)CCCC12CCOCC2 97037,N1(C(CCc2cnc(C)o2)=O)CC2C(CN(C(=O)C(C3CCOCC3)O)C)C2C1 97038,C12(NC(C(C3CCC3)OC)=O)CC(CNC(C3CCN(C)C3C)=O)(C1)OC2(C)C 97039,C1(C(=O)N(C2CCN(C(C3C4CCCC34)=O)CC2)CCO)CC2(C1)CS(=O)(=O)C2 97040,C(C(O)CC(F)(F)F)NC(CC1CN(C(CCOC)=O)C(C)C1)=O 97041,C1(NC(COC(C)C)=O)CCC(N(C(=O)CCNC(=O)OC(C)(C)C)C)CC1 97042,c1(C(=O)NC(CC(C)NC(C=C(C)C(F)F)=O)C)cc(Br)c2[nH]c(C)nc2c1 97043,C(CCC(O)C(=O)N1CCOC(C2CC2)CC1)NC(C1(C)CCSCC1)=O 97044,Cc1c(C(N2CC(CNC(=O)C3=CCCS3)C(C)C2)=O)c(C)n2ccncc12 97045,c1(SCCC)ccc(C(N2CC3(NC(=O)C(C(=O)OC)OC)CC2C3)=O)cc1 97046,c1(C(=O)NCC2CCCC(NC(c3c(OC)nsc3)=O)C2)cccc2sccc12 97047,C1(NC(CC2CC(NC(CC3CC(SC)C3)=O)C2)=O)CC2CC2C1 97048,C1(C(=O)NCc2c(C(=O)NC(c3ncco3)C)occ2)CN(C)C(=O)N1 97049,c1(C(N2CCCC(C(F)F)C2)C(=O)NCc2nccs2)cc2cc(Br)ccc2o1 97050,c1(NC2CC(NC(C(=Cc3cccs3)C)=O)C2)c(C#N)nnc2ccccc12 97051,C(CC(C)(C)C(=O)N1CC(CC(=O)N(C)CC2CC(F)(F)C2)C2(CC2)C1)OC 97052,C1(N(C(c2c(C)nsc2)=O)C)CN(C(c2cn(C3CC3)nc2C)=O)CC12CC2 97053,N1(C(Cc2c(C)ccs2)=O)CCC(C)C(NC(=O)CCOc2ccc(F)cc2)C1 97054,C1(CNC(c2c(CC)onc2)=O)CCCC2(CN(C(c3cnnn3C)=O)C2)O1 97055,C1(N(C(COCCC(C)C)=O)CCO)CCN(C(c2cn(C)nc2CO)=O)CC1 97056,N1(C(C2(CCOCC)CCC2)=O)CCC12CN(C(c1c[nH]c(C(N)=O)c1)=O)C2 97057,c1(C(=O)NC2(c3cnccn3)CCC2)nccc2nc[nH]c12.C12CC1CNC2=O 97058,CC1CC(=O)NCC1C(=O)N(CC(N1CC(CN(C)C)C1)=O)C1CC1 97059,c1(CO)c([N+](=O)[O-])ccc(F)c1Cl.N1(C2c3cn(nn3)C2)CCCC2(CCO2)C1 97060,O=C1CCNc2cc(C(N3CC4C(NC(=O)C(F)(F)C(F)F)C4C3)=O)ccc2N1 97061,N1(C(C2C(C3CN(C(C(CC)OC)=O)C3)C2)=O)CCC2(CNC(=O)N2)C1 97062,C1(CC)C(NC(=O)Cc2c(C)cccc2C)CCCN1C(=O)Cc1ccsc1C 97063,N1(C(CCC=CCC=C)=O)CC(NC(=O)CC(C)c2cnn(C)c2)C(C(F)F)C1 97064,c1(C(N2CCN(C(CN(CC)CC)=O)CC2C(C)C)=O)onc2cc(C)ccc12 97065,N#CCCCCCC(=O)NCCCCNC(=O)Cc1csc(Br)n1 97066,C1(C)(OC)CCN(C(C(C)NC2CCCCC2)=O)C1.C12CCCN(C1)C2=O 97067,c1(C(N2CC=C(C(=O)NC3CC(=O)NCC3)C2)=O)cc2cccnc2[nH]1 97068,C1(NC(=O)CCOCC(F)F)CCN(c2nccn3nnnc23)C12CCC2 97069,Cn1cc(C(N)=O)c(CCCNC2(c3nnnn3C3CCOC3)CCCCC2)n1 97070,CCCCC(O)CC(=O)NC1CN(C(c2c(F)cc(N)cc2F)=O)CC2(CC2)C1 97071,N1(C(C=CC)=O)CC2CCC(C1)N(C(c1cnn(-c3cccc(F)c3)c1N)=O)C2 97072,NC12CCC1CN(C(=O)C(=O)N(CCc1cccs1)Cc1ccc(Cl)cc1)C2 97073,C1(CNC(C2CC(=O)N(C3CC3)C2)=O)CC(O)CN1C(=O)Cc1csc(S)n1 97074,C(=O)(CC(C)(C)C=C)NC(CC=C)CNC(=O)C(c1cccc(F)c1)O 97075,c1(CNC(=O)NC(c2ncc[nH]2)CC)n[nH]c2c1COCC2 97076,O=C1Nc2cccc(-c3ccc(F)c4c3CCC4)c2CO1 97077,C(=O)(C1=CCC(NC(C2CC3CC2CC3O)=O)C1)NCCCC1(C)CC1 97078,N1(C(c2ccc(CNC(CC(C=C)C)=O)nc2)=O)CCC(N(C)C)C(C)C1 97079,c1(C(N(CCN(C(C=C(C)c2ccsc2)=O)C)C)=O)cc(C)n(C)c1C 97080,C(CC)(CC)(CCNC(=O)C(C)c1ccsn1)NC(c1c(CC)cco1)=O 97081,Cc1cc(NC(=O)CCOCCN(C)C(C2(C)CCOC2C)=O)cnc1C 97082,c1(OC)cc(OC)c(C(N2CCC(NC(C3CCC3(F)F)=O)C2C)=O)cn1 97083,C(CCCCC(=O)Nc1cnc(NCc2cncc(Cl)c2)cn1)N(C)C 97084,c1(CC(N2CC(N(C(CC(CCC)O)=O)C)C(O)CC2)=O)cc(F)c(N)cc1F 97085,C(C)(CC(=O)N(CC(C)(C)CNC(c1n[nH]cc1OC(C)=O)=O)C)OC 97086,c1(-c2cccc(OC)c2)[nH]c(=NCC2COCCN2C(C)=O)sc1C 97087,N1(C(C2C(CC)CCCC2)=O)CCC(NC(=O)C(C)CC2CCCC2)C(C)(C)C1 97088,c1(C(=O)NC2(C)CC(NC(C(CO)N(C)C)=O)C2)cccc(F)c1Br 97089,CC1(NC(c2coc(CNC(=O)CCn3cncn3)c2)=O)CCOC1C1CC1 97090,N1(C(C(COC)NC(=O)CNc2ncccn2)=O)CCOC(CN=[N+]=[N-])C1 97091,c1(OC)cc(C(=O)O)ccc1OCC1CCCC(N(C)C)C1 97092,c1(C(N2CCC(C)(NC(CCSC)=O)CC2)=O)ccc2cn(C(F)F)nc2c1 97093,C=CC1CCCN(C(C)=O)C1.c12ccc(cc1Cl)NC(=O)CCCn1cc-2nn1 97094,N1(C(CCCC#N)=O)CCN(C(=O)CC23CC(C2)C3)CC1Cc1cccc(F)c1 97095,c1(CC)sc(C(=O)NCC(C)(C)CNC(c2ccc(C(=O)OC)nc2)=O)cc1C 97096,N1(C(C(C)OC)=O)CCC2(CCC(NC(c3cnc4sc(C)c(C)n34)=O)CC2)C1 97097,CCC(C)CCC(=O)NCCC1CC(NC(c2sccc2OC)=O)C1 97098,C12(CNC(Cn3c(C)nnn3)=O)CCCCC1N(C(c1ccon1)=O)CC2 97099,c1(NCCC2(COC)CC2)cc(NC2CC(CO)C23CCC3)nc(C)n1 97100,C1(NC(C(c2ccccc2)C)=O)COC2(C1)CN(C(c1scnc1C1CC1)=O)C2 97101,N1(C(CC2(C)CN(Cc3ccc(OC)nc3)C2)=O)Cc2cccc(F)c2C1 97102,N1(CC(=O)NCCCCC2CN(C(=O)C(CO)N(C(N)=O)C)C2)C(=O)CCC1=O 97103,C(=O)(C1CCCc2nnn(C)c21)N(CC(C)(C)NC(CCOCC(C)C)=O)C 97104,C(=O)(CCC(=O)NN(C)C)N1C(CN(C(C2C(CN(C)C)C2)=O)C)CCC1 97105,N1(C(c2cc(C(C)(C)O)on2)=O)CCN(C(C2CSCCS2)=O)C2COCC12 97106,c1(C(=O)NC2(C(N(C3CC(N(C)C)C3)C)=O)CCCC2)cncc2ccc(F)cc12 97107,C1(C)(CN(C)C(C2CCOCC2)=O)CCCC1NC(=O)CNC(c1ccoc1)=O 97108,C1(Cn2cc(CC(C)O)nn2)CN(C(c2cnncc2O)=O)CCO1 97109,C1(NC(c2cnc(C)[nH]2)=O)CCCCC1NC(=O)COCCc1cccc(F)c1 97110,CC1CN(C(=O)C(C)N2CCC2)CCN1C(=O)C(C)(F)F 97111,c1(C(=O)NC(C2CCCN2C(C2(C)CC(N(C)C)C2)=O)C)cc(O)cc(O)n1 97112,C(=O)(Nn1cnnc1C)C1CN(C(C(N2CC(C)C2)C)=O)CC1C 97113,c1(C(N2CC(NC(C=CCC)=O)C(SC)C2)=O)c(C)nn(C)c1Cl 97114,N1(C(c2c(C)nn(C)c2)=O)CCOC2CN(C(=O)C(C)(O)c3ccccc3)CC12 97115,C=CC1(C(=O)NCC(C2CC2)N(C)C(c2cccc(F)c2)=O)CCCCC1 97116,c1(CC(=O)NCC2C(NC(c3n(C)ncc3)=O)CCC2)ccc(Cl)cn1 97117,N1(C(c2n(C)cc(OC)c(=O)c2)=O)CC(NC(=O)COC(F)F)C2(CCC2)C1 97118,C1(C(=O)NCCCN(C(=O)C(c2ccc(F)cc2)(F)F)C)CCCC(F)C1 97119,C=CC(C)(C)CC(=O)NCC(O)CC(=O)NC(C1CCCC1O)C 97120,c1(C(=O)NCCNC(c2cnnn2-c2ccccc2)=O)snc(O)c1Cl 97121,c1(C(N2CCC(C)(CCNC(C(CSC)C)=O)C2)=O)ccnc2ccsc12 97122,c1(CNCC(C(C)C)NC)c(F)ccc(Br)c1OCc1ccccc1 97123,C1(NC(c2cccnn2)=O)CCC2(CCCN(C(C3SCCS3)=O)C2)C1 97124,Cc1nc(C(=O)NCC(=O)NC(C(=O)O)C(C)C)[nH]c1C 97125,C1(C(=O)NCC2COCCN(C(=O)CCN3CCC3)C2)CC(=O)C12CCCC2 97126,C12(C(=O)NC3CC(C)(NC(C(CC)n4nccc4C)=O)C3)COCC1C2(F)F 97127,c1(C(NC(=NCCOCC)NC(C2CCCO2)C)C)nc2ccccc2s1 97128,CC1=C(C(=O)N2CCC(NC(=O)C=CCN3CCOCC3)C2)C(=O)OC1(C)C 97129,CC1=NS(=O)(=O)N(C)C=C1C(=O)NCC1C=CC(NC(=O)C(C)CC2CC2)C1 97130,C1(C(N2CC(NC(CSCC)=O)C2)=O)CCC2CCC1O2 97131,C1(CNC(CS(=O)(=O)NCC)=O)CN(C(C2CC(=C3CC3)C2)=O)C(C)(C)C1 97132,c1(CC(n2cc(-c3n(CCOC)ncc3)nn2)C)ccc(C(C)C)cc1 97133,N1(C(C(CC)CC)=O)CC(C)(C)C(NC(=O)CC2CCOC(CC)C2)C(C)(C)C1 97134,CN1CC(N(C)C(C2CCN(C(=O)C3=CCOCC3)C2(C)C)=O)CCC1=O 97135,N1(C(C2(CC)CC2(F)F)=O)CC2CCC1C(NC(c1cc(C)c(O)c(C)c1)=O)C2 97136,c1(C(CCOC)NC(C2(c3ccccc3)CC2(Cl)Cl)=O)ccc(C)cc1 97137,C1(CNC(CN(C(C)C)C)=O)CN(C(=O)C(C)Oc2ccccc2Cl)C(C)(C)C1 97138,c1(C(=O)NC(C2CCOC2)CNC(c2ccc[nH]2)=O)cc2c(s1)CCCC2 97139,c1(C(=O)NCC2CC2NC(C23CCC2CC3)=O)cc2c(s1)CCCC2 97140,C(C(CC(F)(F)F)NC(=O)C(C)Oc1ccccc1F)NC(CCC=C=C)=O 97141,N1(C(C(CCC)OC)=O)CCCN(C(c2nc(C)ccc2OCC)=O)C(C)C1 97142,c1(C(C(=O)NCC(C)N(C(C2CCCO2)=O)CC)(C)C)cccc2ccccc12 97143,c1(C(N2C(C)C(NC(C3CC3C)=O)CC2)=O)cc2c(cc1[N+](=O)[O-])OCCCO2 97144,Cc1cc(N)cnc1C(=O)NC1CC2CC(NC(=O)CC3CCCCO3)C1C2 97145,N1(C(C(C2CCCC2)OCC)=O)CC2CCC1CN2C(=O)C(c1ccccc1)O 97146,c1(C(=O)NC2C=CCN(C(C(CC(C)C)C)=O)C2)cc2cccc(F)c2s1 97147,c1(CC(=O)NCCN(C(=O)OC)C)ccc(C)c(Br)c1 97148,C1(C(=O)NCC(=C)C)(CNC(=O)CCc2conc2C)CCCCC1 97149,c1(C(N2CC(F)CC(NC(C3(C)CC3)=O)C2)=O)ccc2c(c1)OCO2 97150,C1(C(N2CC(NC(C)=O)C2)=O)(OC)CCN(C(=O)C(Cl)Cl)C1 97151,c1(C(=O)NCCCC2N(C(C(CC)=CC)=O)CCCC2)cccc2c1C(=O)CC2 97152,C(=O)(C1Cc2ccc(Cl)cc21)NCC1(O)CCCN(C(C=NOC)=O)C1 97153,CC1(C)CCC(CC(=O)NCC(O)C(=O)NCC2(C(O)C(C)C)CC2)C1 97154,Cc1cc2ccc(C(N3CCC(NC(=O)C(C)C4CC4)C(F)C3)=O)cn2c1 97155,C1(C(C)CNC(=O)CCc2cncn2C)CCN(C(c2ccccc2F)=O)CC1 97156,c1(CN2CC(C(=O)NC(C(CC)C)c3ccccc3)C2)ccc2c(c1)oc(=O)n2C 97157,Cc1nc(CCC(=O)NC2CCN(C(c3ccc(C)n3C)=O)C2C2CC2)[nH]c1C 97158,Cc1ccn2ncc(C(=O)NC3(C)CCCN(C(C4CCSC4)=O)C3)c2n1 97159,c1(C(=O)NC2C(CNC(C(C)OCC(C)C)=O)CC2)cccc2nccnc12 97160,C1(CNC(=O)CC2CCCCC2)CCN(C(C2C3CCCC23)=O)CC1O 97161,N1(C(C=CC(CC)=CC)=O)CCC(NC(c2cc(C)[nH]n2)=O)CC1C 97162,c1(C(N2CCC(C3N(C(=O)OC(C)(C)C)CCC3)C2)=O)ccc(F)c(Cl)c1 97163,Cc1cccc(C(n2cc(-c3cncc(F)c3)nn2)CCO)c1.C(=O)CC1CC1F 97164,C1(CCNC(CC=C=C)=O)CCCN(C(c2cncc(N)n2)=O)CC1 97165,C12(C(=O)NC3(CC#C)CCC3)CCC(CN(C(=O)C(C)(O)C3CCC3)C1)C2 97166,Cc1cc(Cl)c(C(=O)NC2CC(C)N(C(C3CC(CF)C3)=O)C2)s1 97167,c1(C(=O)NCCN(C(=O)COC2CCCC(C)C2)CC)cncc2[nH]ccc12 97168,C1(CC(=O)NC2CC2)CCC(C2CC2)O1.C12CCN(C1)C(=O)N2 97169,CC1CN(C(=O)CSc2ccc(Cl)cc2)CCCN1C(c1cnn(C(F)F)c1)=O 97170,c1(CN2C(=O)NC(C)(c3cccc(I)c3)C2=O)ccc(O)cc1[N+](=O)[O-] 97171,c1(CNC(=O)NC2CC(C)SC2)ccccc1C(F)F 97172,N1(C(c2nc(C(C)(C)C)oc2)=O)CCn2ncc(C(N3CC(F)C(F)C3)=O)c2C1 97173,N1(C(C23CC2C3)=O)CCC2CCC(C1)N2C(c1cc(OC=C)c(N)c([N+](=O)[O-])c1)=O 97174,C1(NC(C(CCOC)C)=O)C2CCN(C(=O)C(C)(C)COC(C)C)CC12 97175,C1(C(=O)NCC2(CN(C)C(c3cc(C#N)cs3)=O)CC2)CCc2ccccc2C1 97176,C1(NC(c2ccoc2)=O)CN(C(=O)Cc2ccns2)CCC12CCOCC2 97177,C1(C(CNC(C(CC)n2ccnc2)=O)C)CCN(C(=O)Cn2nnc(C)n2)CC1 97178,N1(C(c2[nH]ccc2CNC(C2(O)CCOC2)=O)=O)CCC2CCC(C2)C1 97179,c1(CSC)cc(-c2ccc(OCc3nccn3C)cc2)cc(S(N)(=O)=O)c1 97180,C12(C(N(CCO)CC)=O)CC(CO)(CN1C(C1CCCCCCC1)=O)C2 97181,c1(COC2C(=O)N(c3cccc(Cl)c3)CC2)cc(I)c(Cl)cc1Cl 97182,c1(C(=O)NC2C(NC(C(C)OCC#C)=O)CC2)cc(N)ccc1O 97183,CC(CN(C)C(=O)OC(C)(C)C)C(=O)NCC1CCC1NC(c1coc(O)n1)=O 97184,Cc1cc2c(cc1C)C(NC(c1ccc(N3CCN(C)C3=O)cc1)=O)CCS2 97185,C(=O)(C1=C(C)N(C)c2nnnn2C1C)NCCN(C(C(CC)OCC)=O)CC 97186,N1(C(CCCSC)=O)CCOC2CCN(C(C3CCCOC3C)=O)CC12 97187,c1(C(=O)NCC(CC(=O)Nc2c(OC)nn(C)c2)OC)cc(C)cc(O)n1 97188,Cc1cc(Cl)ccc1NC(N1CCN(CC(C)(C)F)CC1)=O 97189,c1(CC(=O)N(CCC(C)NC(C(CC)N(C)C)=O)C)coc2c(C)c(Cl)ccc12 97190,CC1NC(=O)OC12CN(C(=O)CC13CCC1CN(C(=O)CC1(C)CCOCC1)C3)C2 97191,C(CCC(CCC)NC(c1c[nH]nc1-c1ccncc1)=O)NC(COCC#C)=O 97192,C(=O)(C1CCc2nccn21)NC(C(C)C)CNC(c1ccc(C(=O)N(C)C)cc1)=O 97193,C1(NC(c2cncc(OC)c2)=O)CCCN(C(C2CSCC(=O)N2)=O)C1C 97194,Cc1cn2c(n1)C(C)N(C(CC1CCCCC1)C(=O)NC(C)C)CC2 97195,CCC(C)(O)C(=O)NCCC1CN(C(C2(c3nccs3)CC2)=O)CCO1 97196,N1(CC(CC)C(C)C)C(=O)CN(CCCc2nccs2)C1=O 97197,c1(C(N(C)CCNC(C2(CF)CCOCC2)=O)=O)ccc2c(c1)N(C)C(=O)CO2 97198,c1(CCN=C(NCC(=C)F)NCCC(=O)N(C)C)ccc2[nH]ccc2c1 97199,C(=O)(C(CC(C)C)C(C)C)NC(C(=O)NCc1c(OC)ccnc1)CCF 97200,C(=O)(CC(C)(C)C)N1CC(NC(C2CCN(C(CC)=O)C2)=O)(CO)C1.C1(=O)C(C)N1 97201,C12(C(=O)NCC3(F)CCC(CNC(c4ccn(C)c4)=O)C3)CC1COC2(C)C 97202,c1(C(=O)NCC2(C(C)NC(C3C(CC)C3)=O)CC2)cnc(C)o1 97203,c1(CC(=O)NC(C)CNC(C2COC2)=O)ccc2ccncc2c1 97204,N1(C(c2nc(C)oc2C)=O)C2CCC1CC(CNC(=O)C(C)Cc1ccco1)C2 97205,O=C(CC(C(F)F)NC(C1CCOCC1)=O)NCCC1CC(F)(F)C1 97206,Cc1cc(O)ncc1C(=O)NCC=CCNC(c1ccc(SC(F)(F)F)s1)=O 97207,c1(NC(C2C(NC(C=CC=CC)=O)CCCC2)=O)cc(Cl)ccc1I 97208,O=C1CN(CC(=O)NCC2CC2CN(C(=O)CC(O)c2ccccc2)CCl)CCN1 97209,N1(Cc2nc(SC)sc2)CCC(CNc2ccccc2)CC1 97210,CC(CC(=O)N1CCCC1COCc1ccccc1)c1cnn(C)c1 97211,N1(C(C(c2cn(C)nc2)O)=O)CCC2CN(c3ccc(Cl)cc3[N+](=O)[O-])CC2C1 97212,Cc1cc(C(F)(F)F)nc(=NCCc2ccc(CC(C)C)cc2)[nH]1 97213,c1(C(=O)NC(C(=O)NC2C(OC)C3(C2)CCC3)CC(C)C)cccc2cncn12 97214,C(=O)(C1=CCN(C(=O)C(C)(C)C2CCCO2)C1)NC(C)CC1CCCO1 97215,Cc1nsc(N)c1C(=O)NCC1(O)CCN(C(c2ccoc2Cl)=O)C1 97216,CC1C(NC(=O)C(F)C(C)(C)O)CC2CCC1N2C(c1ccsc1Cl)=O 97217,C1(C)(CC)CC(C(=O)NCCCC(CO)NC(=O)Cc2ccoc2)CCO1 97218,CN1CCN(C(=O)CNC(c2ccoc2)=O)CC1CNC(C1CC(C(F)F)C1)=O 97219,C(=O)(CC(F)(F)C(F)(F)F)NCC(C)(C1CC1)NC(CCOCCC)=O 97220,C1(NC(C(N2CCN(C)CC2)C)=O)CC2C(NC(c3cnco3)=O)C2C1 97221,N1(C(c2c(C)cncc2)=O)C2CCC(C2)C1CNC(=O)COCC1CCCCO1 97222,C1(C)(CC(=O)N(C)CCNC(c2csc(C3CC3)n2)=O)CCS(=O)(=O)N1 97223,C(CO)(CO)(CO)NC(C1(CCNC(C(C)C2CCCO2)=O)CC1)=O 97224,N1(c2nc(N3CCC(C(C)O)C3)nc3c2CSC3)CCC2(CC1)CNC(=O)N2 97225,N1(C(C(C)c2cc[nH]n2)=O)C2CCC1CC(CNC(C1(CF)CCC1)=O)C2 97226,N1(c2ncnc(N(C)Cc3cccc(SC)c3)c2C)CCC(C)C(C)(C)C1 97227,C(=O)(CC(F)(F)C(F)F)NCC1N(C(c2ccc(CC)c(Cl)c2)=O)CCC1CC 97228,c1(SC)ccc(O)c(C(=O)NCC2CCCC2NC(C2CC2C(F)F)=O)c1 97229,N1(C(c2c(CNC(C3(CSC)CCC3)=O)n[nH]c2)=O)CCC(O)CC(C)C1 97230,C1(CC(=O)NCC2(COC)CN(C(=O)CCn3ccnc3C)C2)CCCCC1O 97231,C1(CNC(c2c(C)n[nH]c2)=O)C(C)CCCN1C(C1CN2CCN1CC2)=O 97232,C12(C(=O)NCC3(CNC(C=CC(CC)C)=O)CCC3)CCCC1(C(N)=O)C2 97233,c1(C(N2CC3(CC(CNC(=O)C(=O)NC4CC4)C3)C2)=O)cccc2occc12 97234,CCN=c1[nH]c(C(N2CCN(C)CC2CNC(c2c(C)ccn2C)=O)=O)cs1 97235,c1(C(N2CCCC(NC(C(C)N(C)C)=O)(CO)C2)=O)cc(F)cc2nn(C)cc12 97236,c1(C(N2CC3CC3(C(=O)Nc3cnn(CCO)c3)C2)=O)ccc(I)cc1 97237,N1(C(C2(C(F)F)CC(=C)C2)=O)CCOCC(CNC(C2(C(=O)NC)CCC2)=O)C1 97238,C1(NC(c2csc(C)c2N)=O)CC2CCCC(C1)N2C(=O)C(C)(C)CC1CC1 97239,C1(C(N2C(C(N3C(C(C)C)COCC3)=O)CSC2)=O)CCC(C)(O)CC1 97240,N1(C(C(C)C#N)=O)CCC12CN(C(c1cnc(C3CCN(C)CC3)[nH]1)=O)C2 97241,C1(C)(CNC(c2ccc(C)cc2)CCO)CCC2CC2C1 97242,C12(C(=O)NCC(CNC(C3C(CC)C3)=O)C)CC(OC)(C1)C2 97243,C(=O)(C1=CC(O)C(NC(=O)C(C(=O)OCC)OC)C1)N(C1CCCCC1)CC#C 97244,C1(n2c(CCOCCC(C)C)nc(-c3c(C)cccn3)n2)CCCCC1(C)C 97245,c1(C(N2C(C(N3CCC(N(C)C)C3)=O)CC2)=O)ccc(OC(F)(F)F)c(F)c1 97246,CC1(C)C(CNC(=O)CC2(O)CCCC2)CCN1C(c1cc(Cl)on1)=O 97247,CC12CN(C(c3ccc[nH]3)=O)CC1CN(C(C1(C3CCCO3)CCC1)=O)C2 97248,N1(C(c2c(OC)c[nH]n2)=O)CCCC(C)(C(=O)NCCCn2nccn2)C1 97249,c1(NCC2(C(=O)NC(c3cnn(C)c3)C(=O)OC)CC23CCC3)ncncc1I 97250,CC1(C)NC(=O)N(CC(=O)NCC2CCC(NC(=O)CCSC(F)(F)F)C2)C1=O 97251,Cc1cc(NC2CCCOC23CCC3)ncc1S(=O)(=O)NC1CCCSCC1 97252,c1(OCC)cccc(CC(=O)NCC2(OC)CCN(C(c3cc[nH]c3)=O)C2)n1 97253,N1(C(CCC(=C)Br)=O)CC(NC(c2cscc2CC)=O)CCC(O)C1 97254,c1(C(N2CCN(C(c3ccc(OC)cc3)=O)CC2C)=O)cc(N)c(C)cc1Cl 97255,N1(C(C(=O)NCCOCCOC(C)(C)C)=O)CCc2c([nH]c3c(Br)cccc23)C1 97256,c1(OC)c(Cl)cc(C(=O)NC2CC(NC(c3nccc(C)n3)=O)CC2O)nc1Cl 97257,N1(C(CC(C)F)=O)CCN(C(=O)CC2CCC(F)(F)CC2)CC12CCC2 97258,C(=O)(C(CC1CC1)NC(=O)COC1CCN(C(=O)CN(C)C2CC2)C1)OC 97259,C1(NC(C2CC(C)C2)=O)CN(CCCC(C)(C)C)CCC1C 97260,CC1(C(=O)NCC2CCC(F)(CNC(c3ccc(C(N)=O)o3)=O)C2)CCC(=O)N1 97261,Cc1cc(C)c(C(N2CC(C(=O)NCC(O)C(F)(F)F)C(C)C2)=O)cn1 97262,c1(C(N(C)CC2OCCN(C(C3(CC)CCCC3)=O)C2)=O)cc(F)c(O)c(F)c1 97263,C=C=C(C)CC(=O)NCCN(CC(C)O)C(=O)CN(C)C1CC1 97264,c1(N(C(c2n(CC=C)ncc2)=O)C2CC2)cnc2c(c1)CN(S(=O)(=O)CC(C)C)CC2 97265,C1(NC(CCc2cc(OC)no2)=O)(CO)CCN(C(C2COCCO2)=O)C1 97266,N1(C(CCC(N)=O)=O)CC2CCCCN2CC1CNC(=O)CC1(O)CCC1 97267,N1(C(c2cnc(C)s2)=O)CCC(C)(C(=O)NCCC2CCCC2(C)C)C1 97268,C1(CC)(NC(=O)CNC=O)CCN(C(=O)C(C)Cc2ccc(F)cc2F)CC1 97269,N1(C(c2cn(CC=C)nn2)=O)CC(F)(F)CC1C(N1CCNC(=O)C1C)=O 97270,C1(OCCOC(C2(CCC)CC2)=O)CCCN=C1 97271,CC1(C)CC1(C)C(=O)NCC1CC(NC(c2csnc2-c2cccs2)=O)C1 97272,CC(C)C(O)CC(=O)NCC1(NC(c2cccn(C3CCC3)c2=O)=O)CCOC1 97273,N1(C(C=CCOC)=O)CCCC(C)(NC(c2cn3ccsc3n2)=O)C1 97274,C1(CC(=O)NCC(C2CCC2)NC(=O)CCOCCOCCCO)CCOC1 97275,c1(OCC)cccc(N2CCOCC(CNC(c3cnsn3)=O)C2)c1[N+](=O)[O-] 97276,c1(C(=O)NC(c2ccccc2)CNC(C(C)(C)C2CC2)=O)ccc(C2CC2)nc1 97277,C#Cc1ccc(C(=O)N(C2CC(NC(C3(CC(C)C)CCNC3=O)=O)C2)C)cc1 97278,CCC(C)(COC)C(=O)NCC(N1CCN(C(=O)CCC=C(C)C)CC1)C 97279,Cc1cccnc1C(=O)NC1CCCC1n1cc(CCC(C)C)nn1.N 97280,C1(CC2NC(=O)N2)CCCN(CCCc2cn(Cc3sccn3)nn2)C1 97281,N1(c2c(I)cncn2)C2CCC1CN(c1ncnc3n[nH]cc13)C2 97282,c1(CNC(CN(C(C)=O)C)=O)ncccc1CNC(C1CN(C)C1)=O 97283,C1(NC(C(CCC(C)(C)C)NC(Cc2c(C)n(C)cn2)=O)=O)CCNC(=O)CC1 97284,C1(OCCOCCOC(=O)C=Cc2ccco2)CN(C(=O)CS(N)(=O)=O)CCCO1 97285,c1(N(C(c2ccnn2CC)C(=O)NC(CC)C)C)ccc(C)c(F)c1 97286,C1(C2CCN(C(C3CC3OCC)=O)CC2)(NC(C=C(CCC)CCC)=O)CC1 97287,CC1(C)CCC(F)(F)CC1C(=O)NC1CCN(C(=O)CC2CC=CC2)CC1F 97288,C1(CC(=O)NC2CCCC(NC(=O)C=C3CCCCC3)C2)(OC)CCCCC1 97289,C(=O)(C1=COCCO1)NCC1C(NC(c2n[nH]c(C)c2Cl)=O)CCCC1 97290,N1(C(c2c(CCC)nco2)=O)CCCC2CN(C(c3cccc(C)c3)=O)CCC12 97291,CS(=O)(=O)c1ccc(C=CC(N2CC3CN(C(=O)C=CBr)CCC23)=O)o1 97292,c1(-n2c(C(CC(C)C)NCc3n(CC)cnc3)nnn2)ccc(OC)cc1 97293,CON(C(=O)C=CCNC(c1sccc1C#N)=O)C(C)C 97294,C1(c2cn(C3CN(C(C(C)(C)OC(C)=O)=O)C3)nn2)C(C)(C)C1(C)C 97295,N#CC1CCC(CC(=O)NCCCCC(=O)NCCN2CCC(O)CC2)C1 97296,C1(NC(c2scc(C(C)=O)c2)=O)CC(NC(c2cncc(C(F)F)c2)=O)CC1O 97297,C1(C)(CN(C(=O)CC2C=CCC2)C)CCCC1NC(c1sccc1Cl)=O 97298,C(CC(C(=O)N1CC(N2CCCC2=O)C1)NC(=O)Cn1cnnc1)OC 97299,N1(CCC(N2CCCC(NC(C=C(CC)CC)=O)C2)=O)Cc2ccccc2C1=O 97300,c1(NC)ccc(C(N2CC(NC(=O)CCc3ccc(O)nc3)C(F)C2)=O)cc1F 97301,c1(CNC2CCN(C(C(C)OC(C)(C)C)=O)C2)c(I)ccnc1F 97302,N1(C(C23C(C)(C)C(CC2)C3)=O)CC2CCC(CNC(C3CCCS3)=O)C2C1 97303,N(C(=S)NNC(=O)c1cccnc1-c1cn[nH]c1)c1ccc(OC)cc1 97304,c1(OC)ccccc1CNC(C(=O)NCCC(F)(F)F)=O.C1C(O)CNC(=O)CO1 97305,c1(C(N2CCCC(C)(NC(C(C)c3ccsn3)=O)C2)=O)ccc2[nH]ccc2c1 97306,N1(C(CC(C)NCCC(O)C(F)F)=O)CCC(CS(N2CCOCC2)(=O)=O)CC1.CO 97307,C1(C2CC2)(NC(C(COCC)NC(c2cnn(C(F)F)c2)=O)=O)CCC1 97308,c1(CC(=O)N(c2ccc(I)cc2)CCC)cc(OC)cc(=O)[nH]1 97309,C(c1cn[nH]c1)=C(C)C(=O)N1CC(n2cc(CNC(c3cocn3)=O)nn2)C1 97310,C(=O)(C(F)(F)C1=CCOCC1)NCC1(NC(C(=O)NCC(F)F)=O)CC1 97311,N1(C(C)=O)CCCC1C(=O)NCC1(F)CC(NC(C2CC(C)=NO2)=O)C1 97312,C(=O)(C(C)(C)n1cc(NC(=O)C(N2CCC2(C)c2ccccc2)=O)cn1)OCC 97313,c1(C(=O)NCCC2CCN(C(C(COC)O)=O)C2)ccc(OC)c(SC(C)C)c1 97314,c1(C(=O)NC2C(CNC(c3c(C)c[nH]c3)=O)CCCC2)cc(Cl)ncc1Cl 97315,C1(C(=O)NC2(C)CC(=C)C2)CC2(CCN(C(=O)Cc3cc(C)sc3C)C2)CO1 97316,C1(C(N(CCOC)C2CC2)=O)CCCN(C(c2cc(OCC)cnn2)=O)C1 97317,Cc1cnsc1C(N1CCCC1C(C)(C)CNC(=O)Cc1cnn(C)c1)=O 97318,c1(C(=O)NCC2CCCN(C(C(C)OC)=O)C2)ccnc(P(C)(C)=O)c1 97319,c1(NC(C2CC(CNC(c3ccc(C)s3)=O)C2)=O)ccccc1N=[N+]=[N-] 97320,C(=O)(CC(C1CC1)NC(=O)C(O)CNC(C1CCCO1)=O)OC 97321,c1(OC)ccc(C(=O)NCCC2CN(C(C3C(C)(C)C3(C)C)=O)CCO2)nc1N 97322,N1(C(c2c(CC)nn[nH]2)=O)CCOCC1CC(=O)N(C1CCN(C)C1=O)C 97323,c1(C(=O)NCC(C2CC2)NC(c2n(CCC)ncc2)=O)cc(OC)ccc1OC 97324,C1(OC)CN(C(=O)CC(C)SC)CC1NC(=O)CCC1CCCCCC1 97325,N1(C(CN(C(C)C)C)=O)CCN(C(C2CC(C)OC(C)C2)=O)C(CS(C)(=O)=O)C1 97326,n1(CC)ncnc1C(C)NC(=O)C(C)(C1CC1)N(C)C(C1CCC(N(C)C)C1)=O 97327,N1(C(CC2(C)CC2(Cl)Cl)=O)CC2CCC1C1CN(C(=O)CCc3ccon3)CC21 97328,N1(C(=O)CCc2cccc(N3CCCS3(=O)=O)c2)CCC(O)C12CCSC2 97329,C(=O)(C1CCCc2nnn(C)c21)NCC1CN(C(c2nccc(C)n2)=O)CC1C 97330,N1(C(c2c(CC)ocn2)=O)CC(C(=O)NCC2CCCC23CCC3)C(F)(F)C1 97331,N1(C(C(CC(CC)C)C)=O)CCC2(CC1)CCN(C(=O)C(C)(C)C1CCCO1)C2 97332,C1(C(N2CCCC(CN(C(=O)CCF)CC)C2)=O)CCC2(CCC2)CO1 97333,c1(C(=O)NC2CCN(C(COCCC(C)C)=O)CC2F)cc2cc(Cl)ccc2s1 97334,C(=O)(CC1=NN(C)C(=O)C1)NC12CC(CNC(C(CC=C)(C)C)=O)(OC1)C2 97335,S(=O)(=O)(c1ccc(N2CCC(n3cc(Cl)cn3)C2)c(Br)c1)N(C(COC)OC)C1CC1 97336,N1(C(C2C(=C)C2)=O)CC2CCCC(CNC(c3c(CC)noc3C)=O)C2C1 97337,Cc1cccc(C(C(C)C)NC(=O)NCCc2nc(C(C)(C)C)no2)c1 97338,C1(CNC(Cc2nc(C)sc2)=O)CCC(C)CN1C(=O)C=Cc1cnn(C)c1 97339,CCC(CC(C)C)C(=O)NCC1CCCC1C(=O)NC1(C(=O)OC)CC1 97340,N1(C(c2cc(C)no2)=O)CCCC(C(=O)NCC23CCCC2C3)C1 97341,C1(CNC(C(CC)OC)=O)CN(C)CCN1C(=O)CCOCC(C)C 97342,c1(OC)ccc(C(N2CCC(NC(c3cnc(C)nc3C)=O)C2)=O)cc1OC 97343,Cc1ccc(F)c(OCC(N2CC3CCC2C3NC(C2CC3CC3C2)=O)=O)c1 97344,Nc1cc(C(N2CCN(C(=O)Cc3cncnc3)C3CC23)=O)c(F)c(F)c1F 97345,C1(C(=O)NCCCNC(=O)Cc2cncnc2O)CCC12CCOCC2 97346,C1(CNC(c2cc(CO)[nH]n2)=O)C2CN(C(=O)C=CC3CCC3)CC12 97347,N1(C(C2CCN(OC)CC2)=O)CCC2CN(C(=O)C(O)C(F)(F)F)C(C)C12 97348,C1(CC#C)(C(N2CC(O)C(O)C2)=O)CCN(C(c2cc(CC)oc2C)=O)C1 97349,N1(C(C(C)NC(N)=O)=O)CC(NC(=O)C(F)(F)c2nccs2)C(C)C1 97350,C1(OC)(CNC(C2CC(O)C2)=O)CN(C(C2(c3ccccc3)CC2(Cl)Cl)=O)C1 97351,CCC(CC)C(=O)NCCN(C(c1nnsc1SC)=O)C1CC1 97352,c1(N(CC=C)C)nc(N2CCCC(C(N)=O)C2)c2c(n1)CCCCCC2 97353,c1(C(=O)NCC(CC)(C)NC(=O)CCCSC)cnc2ncccn12 97354,C1(CCC(=O)N(CCNC(CNC(N)=O)=O)C2CC2)CCCC(O)C1 97355,C(C(N)CCC(C)(C)C)OCC.N12CCCC(C1)Cc1nc(sc1)C2 97356,c1(C(N(C)CC2CN(C(C3CC(N=[N+]=[N-])C3)=O)CCO2)=O)ccn2nccc2n1 97357,c12ccc(c(F)c1)[nH]2.C1(C(=O)NCCC#C)C2CN(C(=O)OC)CC12 97358,c1(C(=O)NC2(CCCC(=O)N(CC(=O)NC3CC3)C)CCC2)ccc(F)cc1F 97359,CCCCC(CC)CC1C(=O)NC2CCN1C2.C1(C(=O)OC)(COC)CCOCC1 97360,CC(CC(C)(C)C)C(=O)N1CC(NC(=O)C(C)(C)Cc2ccc(O)cc2)C(C)C1 97361,c12ccc(cc1O)c(=O)n2C.C(c1ccccc1)=CCSc1nc(C)on1 97362,c1(C(=O)NCC2CCC2NC(CCSCCC)=O)c(F)cccc1F.C(C(=O)OC)N 97363,C1(N(C(C(CSCC)NC(C2CC(=O)C2)=O)=O)C)CCCC(C)C1C 97364,c1(C(=O)NCC(CCNC(CN(CCC)C)=O)O)c(F)c(F)cc(F)c1F 97365,CC(C)P(=O)(CC(=O)NCC(CNC(=O)CCCF)CO)C(C)C 97366,C1(C(N2C(CN(C(CC(C)N(C)C)=O)C)CCCC2)=O)CNC(=O)CC1(C)C 97367,C1(C(N(CC(O)CNC(=O)CNC(c2cccnc2)=O)C)=O)COCCN1C=O 97368,C1(O)(CNC(=O)COCCOc2ccccc2)CCCN(C(=O)C(F)=C2CC2)C1 97369,Cc1ccccc1OCCCC(=O)NC1CCCC1NC(C1(O)CC(CF)C1)=O 97370,N1(C(CCCC(=O)NCC)=O)CC(NC(c2noc(C3CC3)c2C)=O)CC12CCC2 97371,N1(C(C(CC)NC(C)=O)=O)CC(C)C(N=c2[nH]n(C(C)C)cc2[N+](=O)[O-])C1 97372,C(C(C)(C)C(=O)N(C)CCN(C)C(N)=O)N(C(=O)C=C1CCCCC1)C 97373,Cc1cccc(CC(=O)NCC2CCCN(C(C3CC(O)(C(F)(F)F)C3)=O)C2)c1 97374,c1(C(N2CC(OCCNC(C(CC=C)OC)=O)C2)=O)cc2n(n1)CCCN2 97375,CCCC(CNC(c1cc(Cl)n(C)n1)=O)C(=O)NCC1(CCOC)CC1 97376,Cc1ccc(C(O)Cc2cn(C(C)C(=O)N(C)CCN3CCCC3)nn2)cc1 97377,N1(C(C=CCC)=O)CCCC1C(C)(C)CNC(C1CC(O)C1)=O 97378,C#CCC(C(=O)NC)NC(c1coc(CNC(=O)CSC2CC2)c1)=O 97379,c1(CC(N2CCC(NC(c3ncc(F)cc3Cl)=O)C2)=O)cc(Cl)cc(Cl)c1 97380,N1(C(CC=CC=C)=O)CC2(CCN(C(c3sccc3Cl)=O)CC2)CC1C 97381,C1(CNC(=O)CCOC2COC2)(NC(c2cc[n+]([O-])cc2)=O)CCOCC1 97382,Cc1cn(C)nc1C(N1CC(O)(CCc2cn(CCc3ccccc3)nn2)C1)=O 97383,C1(CC)CN(C(=O)CN(C)C(C2(C#N)CC2)=O)CCN1C(=O)COc1ccsn1 97384,c1(CC)ccc(C(N2CCOCC2CNC(=O)CC(C)COC)=O)nc1 97385,C1(CC(=O)NC(C)C(C)(C)NC(c2cccc(C(F)(F)F)c2)=O)CCC(=O)N1C 97386,N1(C(c2nccc(C)c2)=O)CCN(C(c2cnc3[nH]cncc2-3)=O)C2CCC12 97387,Cc1nccn2ncc(C(=O)NC3CC3NC(=O)COC3(C)CCOCC3)c12 97388,c1(C(=O)NC(CNC(c2c(C)nc(OC)s2)=O)C)cnc(O)c(C(F)(F)F)c1 97389,c1(C(=O)OCC)cnc(N2CCN(c3ccnc(C)n3)C3CC23)nc1C 97390,c1(C(N(CCC)CCNC(C2CC(C(C)C)C2)=O)=O)ccncc1N=[N+]=[N-] 97391,C1(CC(=O)NCCOC2CCN(C(c3c(C)cno3)=O)C2)CCC(C)(C)CC1 97392,c1(C(=O)NC2CCN(C(c3cc(OC)cc(Cl)c3)=O)C2C)cccc2cnnn12 97393,c1(C(=O)OCC2CC2C2CCCO2)cnn2ccsc12 97394,O=C(C1CCCc2nn[nH]c21)N1CCC2(CCCN2C(C2CCC(F)C2)=O)C1 97395,N1(C(C(C=C)C)=O)CC2CCCC(N(C)C(c3nnsc3CC)=O)C2C1 97396,N1(C(C(CC)COC)=O)CCCC(F)(CNC(=O)CSCc2cccc(Cl)c2)C1 97397,CC1CN(C(C2CC2(Cl)Cl)=O)CC1CCNC(C1CCCCCC1)=O 97398,c1(OC)ncc(C(=O)NCC(C2CC2)NC(=O)CCNC(C2CCCCC2)=O)s1 97399,c1(C(C)C)nccn1CC(=O)N(C)CCN(C(=O)CN1CCC1C)C(C)C 97400,C1(CC(N2CCC(C)(CCC)C2)=O)CC2(C1)CN(C(C1(C)CNC(=O)N1)=O)C2 97401,C(=O)(CCCCCF)NCC(C)(C)NC(C(C(=O)N(C)C)C1CC1)=O 97402,c1(OCCC(C)NCCS(N)(=O)=O)ccccn1 97403,CC(C(=O)OC(C)(C)C)C(=O)Nc1ccsn1.C12(C)CN(C1)C(=O)CO2 97404,C(CC(C)C(=O)N1CC(NC(c2sc(C)cc2C)=O)C(CO)C1)OC 97405,c1(CN(C)CC2CCN(C(=O)COCc3cccc(Cl)c3)C2)ncccc1F 97406,c1(C(C(=O)NC2CCCC2)O)ccc([N+](=O)[O-])cc1.C1(COC(=O)CNC=O)CC(N)C1 97407,c1(NC(C(CC)n2cnc(-c3nn[nH]n3)n2)=O)ccc(Br)c2c1CCO2 97408,C=C(C)C1CN(C(c2cc(CCNC(=O)C(C)(C)N(C)C)on2)=O)CCO1 97409,c1(OC)cc(OC)nc(N2CC(CO)(NC(=O)C(O)C(C)C)C2)n1 97410,C(CC(C)C)(C(=O)NCC(n1ccnn1)C)ONC(c1c(CC)ncs1)=O 97411,c1(OC)ccc(C=NO)cc1NCc1ccc(OC(C)C)cn1 97412,CC1CCCC1(C)C(N1CCOC(CNC(=O)Cn2cc(N)cn2)C1)=O 97413,CC1(C)CCCC(CCN(C(c2ncc(Cl)s2)C(=O)NCCCOC2CC2)C)C1 97414,C1(CNC(CCn2c(C)ncc2)=O)CCN(C(=O)CCc2cncnc2)CC1O 97415,CCCCC(O)C(=O)N1CCN(C(c2cc(OC)cc(F)c2)=O)C(CCC)C1 97416,C1(NC(COCc2nnc(C)s2)=O)CCN(CCc2ccc(F)c(F)c2)CC1C 97417,CC(CN=c1[nH]c(=NCc2ccccc2CCO)[nH]c2c1CCCC2)CC(C)O 97418,C1(CC)CCCCC1C(N1CCCCC1CCNC(C1(C)CC1C(F)(F)F)=O)=O 97419,C1(NC(=O)Cc2ccco2)COCCN(C(C2CCN(C3CC3)C2=O)=O)C1 97420,C#Cc1cc(NC(=O)C(C2CCCO2)NC(=O)Cc2csnn2)cc(F)c1 97421,c1(OC)ncc(C(=O)NC(C)C(CO)NC(c2ccc(F)cc2SC)=O)cc1C 97422,c1(CCC(=O)N(CCNC(C(C)(C)OC(C)=O)=O)C)ccc(Br)nc1 97423,c1(N2CC3(CN(C(=O)C=Cc4ccc(Cl)nc4)C3)C2)ncnc2ccc(Cl)cc12 97424,c1(OC)cccc(CC(N2CCOC2=O)=O)c1.C1(C)C(=O)N1 97425,C1(C(N(CCNC(c2ccc(CC)cc2F)=O)C)=O)CC(=O)N(C)C(=O)N1 97426,Cc1ccc(C(N2CCN(C(C3(c4cccc(F)c4)CC3)=O)C3CC23)=O)cc1Cl 97427,Cc1cc(C(=O)NCC(C)(Cn2cccn2)NC(C2CN(C)C2)=O)n[nH]1 97428,CCC(C)CC(=O)NC(c1ccc(COC)s1)C(=O)N(C)C(c1cccc(C)c1)C 97429,C1(C(N2CCN(C(C(=O)NCC3CC3)=O)CC(CO)C2)=O)CCc2nnnn2C1 97430,c1(OC)cc(CC(N2CCC(NC(C3CC3C)=O)C2(C)C)=O)ccc1Cl 97431,C(=O)(C(CCc1ccccc1)N1CCOC(CN(C)CC2CC2)C1)NCCOC 97432,N1(C(c2cc3nccnc3cc2Cl)=O)Cc2cc(Br)ccc2CC1C.CC(=O)O 97433,N1(C2CN(C(c3cnc(C)o3)=O)C2)CC(NC(C2CCC3CC23)=O)CC1=O 97434,c1(C(N2CC(CC)C(NC(=O)COC3CC=CC3)CC2)=O)cc2cccnc2s1 97435,c1(NC2(C)CC(NC(N3C(C(=O)OC)CC3)=O)C2)cccc(S(=O)(=O)N(C)C)c1 97436,Cc1ncn(C)c1C(=O)NC1(CO)CN(C(=O)CSc2ccc(Cl)cc2)C1 97437,C1(C(=O)NC(c2ccc(SC)cc2)C)CCN(CC2CCCN(C)C2)CC1O 97438,C12(C(=O)NC3CC(C(C)NC(c4cnc(C5CC5)o4)=O)C3)CCCN1CCC2 97439,N1(C(c2cnc(C3CCCCC3)s2)C(=O)NC(CC)C)CCC(O)CC(C)(C)C1 97440,Cc1nc(NCCC2=CCCC2)cc(N2CCCN(S(C)(=O)=O)CC2)n1 97441,c1(NCC(C2(O)CN(C(CCCSCC)=O)C2)(C)C)ncc(C)cc1[N+](=O)[O-] 97442,C=C(CNC(=O)CSCCNC(=O)CC(CC)C1CC1)C(F)(F)F 97443,C(C(=O)Nc1nonc1C)(C(C)C)NC(C1C(C)(CC)C1)=O 97444,C=C=C(C)CC(=O)NCCN(CC(C)O)C(=O)CC1CC(OC)C1 97445,C(Cc1ccoc1)(C(=O)N(CC(C)(C)N(C)C)C)NC(C1C(CC(C)C)C1)=O 97446,Cc1cc(Br)ccc1CC(=O)NC1CC1NC(C1(C)CC(C)(C)C1)=O 97447,CCCC(C)(O)CC(=O)NC(c1ccc(C(C)C)cc1)CNC(=O)C(F)CC 97448,Cc1cc([N+](=O)[O-])cc([N+](=O)[O-])c1NC(C)CNC(c1n[nH]cc1Cl)=O 97449,CC(C)C(C)CC(=O)NC1CN(C(=O)CN2CC3CCC2C3)C1 97450,c1(C(=O)NC2CCCC2C(=O)Nc2ccc(Cl)cc2Br)c(Br)cccc1[N+](=O)[O-] 97451,c1(C(N2C(CNC(CC)=O)CC(C(F)(F)F)C2)=O)cc2c(cc1F)NC(=O)CC2 97452,c1(C(C)(O)CNC(=O)C(N)c2ccoc2)cccc(I)c1 97453,CCC(C)CC(C(=O)NC1CC1)NC(c1cnn(C2CC2)c1)=O.C1C(=O)N1C 97454,c1(C(=O)OC)cc(-c2cc(C(=O)N=c3[nH][nH]cc3C)ccn2)cc2c[nH]nc12 97455,CC(C)C(C)CC(=O)N(C1CC(C(=O)NCC(O)(C2CC2)C2CC2)C1)C 97456,c1(COC)nc(NCC2CN(C(C)C)C2)cc(=NCc2ccc(CO)c(F)c2)[nH]1 97457,Cc1ccc(C(N2CCOC(C)(CNC(=O)CCc3scnc3C)C2)=O)cc1Cl 97458,CC(CN(C)C)CCC(=O)NCCN(C)C(C1CCC(F)(F)C1O)=O 97459,C(CC(C)(C)C)(C(=O)NC(C)(CNC(=O)CSc1cnn(C)c1)CC(C)C)OC 97460,C1(C2(O)CCN(C(C3CC(CC(F)(F)F)C3)=O)CC2)(NC(CCC)=O)CC1 97461,C(C)(CC(C)(C)C)(c1nnnn1C1COC1)NC1CCC(CC)CC1 97462,c1(C(=O)NCCN(C)C(c2ccc(Cl)c(Cl)c2)=O)cc2sccc2[nH]1 97463,c1(-c2cccc(CNC(CC)=O)c2)nc2c(s1)CCN(C(C1CNC(=O)C1)=O)C2 97464,C1(C(N2CCC(OCCNC(C3(C4CC4)CCCO3)=O)C2)=O)(CC)CCOCC1 97465,Cc1cc(=NC2CCCn3ccnc32)[nH]c(N2CCC(C)C2)n1 97466,N1(C(c2c(C)cccc2)=O)CCN(C(=O)COCc2nc[nH]n2)CCC1C 97467,C1(C(=O)NC(CNC(Cn2cnc(C(C)=O)n2)=O)C(C)(C)C)CCCC2(CC2)C1 97468,C#Cc1cccc(C(N2CC=CCC2C(N2CCCC(C(C)(C)C)C2)=O)=O)c1C 97469,Cc1cnn(C)c1C(=O)NCC(CC(=O)NC(C)(C)CC(C)C)C1CCC1 97470,c1(C(N2C(CC=C)(C(=O)NCC3CC(F)(F)C3)CCC2)=O)cc(C)cc(C#N)c1 97471,c1(C(=O)NC(C)C(C)NC(=O)CCNC(C2CCC2)=O)ccc2ncccc2c1 97472,c1(C(N2CCC(CNC(c3ccc(CO)o3)=O)C2)=O)snc(Cl)c1Cl 97473,c1(C(=O)NC(C(C)C)CCN(C)C(c2cccc(O)n2)=O)ccc2c(c1)CCOC2 97474,C1(NC(c2cc(C)nc(O)n2)=O)C2CCCCN(C(=O)Cc3c[nH]nc3C)C12 97475,C(=O)(C1=C2CCN=C2NC=C1)NCC(CNC(C1N(C)CC(C)(C)C1)=O)O 97476,C(=O)(C1=COCCC1)N1C(C)CC(NC(C2CNC(=O)O2)=O)C1 97477,C(=O)(C1OCCn2ccnc21)N(CCCCNC(C1(C(=O)NC)CCC1)=O)C 97478,C1(CNC(Cn2c(C)ccn2)=O)CCC2CN(C(=O)CCc3nncs3)CC12 97479,c1(-c2onc(-c3cccc(OC)c3)n2)cccc2cc(OC)ccc12 97480,C12(NC(CSCCOC)=O)CCC(C1)N(C(c1cccc(-n3ccnn3)c1)=O)C2 97481,CC(F)(F)CCCC(=O)NC1CC(F)CN(C(c2c(F)cccc2Br)=O)C1 97482,CC1=C(C(=O)NCCCOCCN(C(=O)C(C)(C)C2CCOC2)C)COCC1 97483,C1(C(N2C3C(CNC(C(C(C)O)C)=O)CC(CC3)C2)=O)CCc2cnn(C)c2C1 97484,N1(C(C(C)(C)O)=O)CC2CCC1CN2C(C1(C#N)CCC1)=O 97485,C1(C(=O)NC(CCCNC(c2c(Cl)cc(C)s2)=O)C)CCCC2(CCC2)O1 97486,C1(C)(C(=O)NC23CC(NC(CCSC)=O)(C2)C3)C2CCC(C2)C1(C)C 97487,N(C1C(=O)Nc2ccc(F)cc21)C(C1=C(C)OCC1)=O 97488,N1(C(C(N2C(C)CN(c3ccncc3)CC2)=O)=O)CCC(C2(O)CCC2)CC1 97489,CN1CCC1C(N1CCC1C(N1CC(C(C)(C)C#N)C1)=O)=O 97490,CCC(C(=O)OC)C(=O)N1CC(CO)(NC(=O)C=CC2CCCCC2)C1 97491,c1(C(=O)Nc2cccc(NC(C3(SCC)CC3)=O)c2)sccc1S(N)(=O)=O 97492,C(=O)(C1CC(C)(C)Oc2ccccc21)N1CCC(NC(c2n(C)cnc2)=O)C1 97493,N1(C(C(=O)NCC(c2cn(C)nc2)(F)F)=O)CCc2c(ncn(C)c2=O)C1 97494,O=C(C1CCCn2cncc21)NC1CCN(C(C2CCCCC2O)=O)C1 97495,Clc1ccc(-c2nc(CN3CC4CC4C3)n(-c3cccnc3)n2)cc1Cl 97496,N1(C(C2(COC(C)C)CC2)=O)CC(N(C(=O)C(C)CN2CCOCC2)C)C(O)C1 97497,Cc1ccc(C(=O)NC23CC2CN(C(c2ncn(C)n2)=O)C3)c2ccccc12 97498,c1(C(N2C(CNC(C(COC)C)=O)CCCCC2)=O)cnn2c(Cl)cccc12 97499,c1(C(=O)NCC2COCCN2C(c2ccnnc2O)=O)c[nH]c2ncnc(O)c12 97500,Cc1ccc([N+](=O)[O-])cc1C(N1CC(O)CC1C(=O)Nc1cnc(Br)c(Cl)c1)=O 97501,C1(C(=O)NCC2CC(NC(COC(C)(C)C)=O)C2)CCC(n2cccc2)CC1 97502,c1(C(=O)NCC(CC)(C)NC(C2CCC23CCC3)=O)nsc2ccccc12 97503,Cc1[nH]nc(C(=O)NC2CN(C(=O)C=CCF)CC2C(F)F)c1C 97504,N1(C(C(C(=O)OCC)(C)C)=O)CCc2ccccc2C(NC(=O)CCC2CC2)C1 97505,CON(C(=O)C=CC(C)NC(=O)C(C(C)C)NC=O)C1CCC1 97506,CC1(C)CCOC1CC(N1CCCCC1C1CCN(C(=O)C(O)C2CCC2)C1)=O 97507,C(=O)(CC(O)CC(C)C)NCC(C1CCCCC1)NC(C(CC)(CO)OC)=O 97508,N1(C(CC(C=C)C)=O)CCC2CCCC12C(=O)NCCCC(=C)Cl 97509,C(=O)(C1=NOC(C)(C)C1)N1CCCC(CC)C1C(N1CCC1C(N)=O)=O 97510,Cc1cc(C(N2CCCN(C(=O)CCN3CCC3)CC2C)=O)cc2c1CCC2 97511,CCC(C)(C(=O)NC(C1CCN(C(=O)C(C)=CC2CC2)CC1)C)C(N)=O 97512,Cc1noc(C)c1C(C)C(=O)NCC#CCNC(=O)Cc1ccccc1F 97513,c1(C(=O)NC(CCCC)CNC(=O)CC(C)n2cccn2)cc(C)c(C)c(Br)c1 97514,c1(NCC(C)N(C)C(C2CC=CCO2)=O)cc2nn[nH]c2cc1[N+](=O)[O-] 97515,N1(CCNC(C2CC(C3CC3)C2)=O)CCN(C(=O)C(O)C2CCC2)CC1 97516,C1(C(=O)OCC)CCCC(NCCc2ccc(Cl)s2)CC1 97517,c1(OC)cc(C(N2CCC(CO)(NC(=O)CN(C)C)C2)=O)cc(F)c1F 97518,C1(NC(C2(CC=C)CCCC2)=O)CC2CCC(C1F)N2C(=O)CC1CC1CC 97519,c1(CC)c(C(N2CC(C(=O)Nc3cnn(CC)c3)C2)=O)cnn1CO.C(C)(=O)OC 97520,c1(C(C(=O)NCCC(CNC(C(C)(C)OCC)=O)O)CC)c(C)noc1C 97521,C(C)(CO)(C(F)(F)F)NC(C(C)N(C(C(COCC)C)=O)C1CC1)=O 97522,Cc1cc(Cl)cc(Br)c1NC(C1CC(C)CN1C(c1cnc(O)cc1O)=O)=O 97523,C(=O)(CS(N)(=O)=O)N(CC(CCN(C1CCOC1)C(=O)NC(N)=O)O)C(C)(C)C 97524,N1(C(c2ccc(C(N)=O)s2)=O)CCC2CN(C(C3CC(C(F)F)C3)=O)CC12 97525,N1(C(C2(C)CC2(Cl)Cl)=O)CCC(C)(NC(=O)CN2CCS(=O)CC2)C1 97526,c1(C(C(=O)NCc2ccco2)N(CCC)CCC)ncc(CC)[nH]1 97527,CCC(C)(O)C(=O)NCCC1CCCN1C(=O)CCOC(C)C 97528,C12(C(=O)NCCC(C=C)C)CC(CN1C(=O)CC1COCC1O)C2 97529,C(=O)(C1CCCc2nncn21)N1C(CNC(C(C)S(N)(=O)=O)=O)CCC1 97530,n1(CCC)cc(C(=O)NCC2CCCC2NC(=O)C(C)SC(F)(F)F)cn1 97531,c1(C(=O)NCCN2CCC(O)C(O)C2)c(Cl)cc(F)cc1Cl 97532,c1(SCn2cc(C3C(C)CCN3C(=O)OC(C)(C)C)nn2)cc(O)nc(O)n1 97533,c1(C(=O)NCC2(F)CC(NC(C3ON=C(C)C3)=O)C2)ccccc1CC#N 97534,c1(C(=O)C2CC2c2ccccc2)ncn(Cc2cc(C(F)F)no2)n1 97535,C1(C(=O)NCC(C)(C2CCC2)NC(C=COCC)=O)CC2(C1)CC(O)C2 97536,CCCCC(CNC(C1OC(C)CC1C)=O)NC(=O)C(C)CSC 97537,CC1=C(C(=O)N2CCC(NC(C3CCCC(F)(F)C3)=O)C(F)C2)C(=O)OC1(C)C 97538,N=c1[nH]c(=NCC2CCOCC23CCCC3)[nH]c(=NCCn2ccnc2)[nH]1 97539,c1(C(=O)NCC2CCCN(C(C3CC3F)=O)C2)ccc2c(O)nnc(O)c2c1 97540,CC(C(=O)NCC1(F)CN(C(c2ccc(Cl)cc2O)=O)C1)C1=CCCC1 97541,c1(C(N2C(C(N3CCCC(C)CC3)=O)CC2)=O)ccc(C#N)cc1Cl 97542,Cc1cc(CC(=O)N(CC(O)CN(C)C(C2(O)CCCC2)=O)C)ccn1 97543,CCC(CCC(=O)NCCF)NC(C1CCC(=O)NC1)=O 97544,Cc1nc(C(=O)N(CCNC(=O)Cc2cn(C3CC3)cn2)C(C)C)c(C)s1 97545,S(=O)(=O)(c1ccc(C(N2CCCC2C(N2CCCC(F)C2)=O)=O)cc1)NC 97546,CCCCCC(F)C(=O)N(C(C)C(N1CCOC2(CC2)C1)=O)C 97547,N1(C(C=C(CC)CC)=O)CC(C)OC2(CCN(c3nnc(-c4ccon4)s3)CC2)C1 97548,N1(C(C2CC(=C)C2)=O)CC2CC(C1)CN(C(=O)COC1CCC1)C2 97549,C1(C(=O)NC(CCO)C2CCC2)C2CCC(C2)N1C(=O)CC1CSCCO1 97550,N1(C(C(=O)N(c2ccccc2C)C(CC)C2CC2)=O)CCCC(C)(CC#N)C1 97551,N1(C(CC2CCN(C(C(C)CC3CCCC3)=O)C2)=O)CCC2(CCCCC2)C1 97552,c1(OC)ccc(C=CC(=O)NCC2CCCCN2C(c2csc(C)c2)=O)cc1Cl 97553,C(CC(O)C(=O)N=c1ccn(C2CC2)[nH]1)NC(=O)C=CC1CCOCC1 97554,c1(NCC(N2CC(NC(=O)OCC)C2)=O)cc2c(s1)CCC2CN 97555,C(=O)(C1=NOC(C(C)(C)C)C1)N1CC(CC(C)NC(c2ccc(CF)cc2)=O)C1 97556,c1(N2CCN(C(=O)NCCC(CC)CO)CC2)cc(OC)c(OC)c(F)c1 97557,C(=O)(CCCCC(F)(F)F)N(C)CC1CCCC(NC(COCCSC)=O)C1 97558,C1(N(C(C(CC)CC(C)C)=O)C)CCCC2CN(C(c3csc(=N)[nH]3)=O)CC12 97559,c1(C(C)C(=O)NC2CN(S(C)(=O)=O)CC2CC(=O)O)ccc2ncccc2c1 97560,C(=O)(C(C)C(C)C(C)(C)C)N1CC(CCNC(c2c(OC)cc(F)cc2)=O)C1 97561,CC1(C)CC(CC(=O)NC23CC(CNC(C4C5CCC(F)(F)C45)=O)(C2)C3)C(=O)O1 97562,CC(C)(CNC(=O)CC1CCCN(C(c2cccc(=O)o2)=O)CC1)CN=[N+]=[N-] 97563,N1(C(c2cn(CC(C)O)c(=O)cc2)=O)CCC2CN(C(C3(O)CCOC3)=O)CC12 97564,N1(C(CSc2ccc(C)cc2)=O)CCC(NC(=O)CN2CC(C)C2)CC1C 97565,c1(CC(=O)N(CCCNC(CC(C)OC)=O)C)cccc(OC(F)F)n1 97566,c1(CNC2(c3ccc(C)cc3)CCOCC2)ccc2c(c1)NC(=O)NC2 97567,C1(NC(C(=O)N(C)C)=O)CCCCN(C(c2c(N)cncc2Br)=O)C1 97568,c1(N(CCCN(C(=O)COC(F)(F)F)C)C)cc2c(cn1)C(=O)CCC2 97569,C1(CNC(COCC)=O)CCN(C(C2(c3c(Cl)cccc3Cl)CCC2)=O)CC1C 97570,CC1CN(C(c2cncs2)=O)CC2(CCN(C(=O)CSCc3ncc[nH]3)C2)O1 97571,Cc1cc(C(=O)NCCN(C(C2CCC(=O)NC2)=O)C(C)C)cc(C)c1O 97572,C1(C(=O)NCC(C)(O)CO)C2CN(C(=O)Cn3nccn3)CC12 97573,C1(C(N2C(CNC(c3c[nH]cc(Cl)c3=O)=O)CC2)=O)OC2CCC1CC2 97574,N1(C(COCC=C)=O)CC2(CNC(=O)Cc3csc(C(C)C)n3)CC1(COC)C2 97575,c1(N(C(CC(CC)C)=O)C2CNCC2C#N)nc(-c2ccccc2)cc(C)n1 97576,C=C(C)CCCC(=O)N1CC(C(=O)NC(C)CCCCCC)OC(C)C1 97577,C1(C(N(c2cc(C)no2)C)=O)CCC2(CN(NCc3csc(N(C)C)n3)C2)O1 97578,CC(C)(CCNC(c1ccc(NC=O)cc1)=O)CN=c1[nH]c2cc(Br)cnc2s1 97579,C1(NC(CC2N(CC)CCC2)=O)CN(C(c2ccc(N)cc2O)=O)CC12CCC2 97580,C1(C(N2C(CCNC(C(C3CCCCC3)OC)=O)CCC2)=O)CCCC1C1CC1 97581,N1(C(c2[nH]cc(CC)c2)=O)CC2(C1)CN(c1nc(SC)ns1)C2 97582,Cn1cnc(CC(O)C(=O)NCC(C)(C)NC(=O)CCc2cnco2)c1 97583,C(CN=c1[nH]n(C)cc1[N+](=O)[O-])C1CCC(CNC(C23CCC(CC2)C3)C)CC1 97584,c1(C(=O)NCc2cc(C(N(C(CO)C3CC3)C)=O)sc2)cnn(C)c1Cl 97585,C(=O)(CCCC(=O)N1CCOCC1C(=O)NCC1(C)CC(O)C1)OCC 97586,c1(C(=O)NCC2CN(C(CN(C)S(N)(=O)=O)=O)C2)cc2n(n1)CCCCO2 97587,C(=O)(C(O)CC(C)C)N1C2C(NC(CC(CC)OC)=O)C(C2)C1 97588,CC(=O)C(C(C)C)NC(=O)CN(C(=O)C(C)Oc1cccnc1)C(C)C 97589,c1(C(N2CC(C(C)NC(c3cccn3C)=O)C2)=O)ccc(Br)cc1O 97590,c1(C(C)C)nnc(C=CC(=O)NCCC2(CNC(C3CC4(C3)CC4F)=O)CC2)o1 97591,O=C1COc2cc(C(N3CCN(Cc4ccc(F)cn4)CC3)=O)ccc2N1 97592,c1(C(C)=O)cc(=NCCC2CCC(NC(=O)C(N)=O)C2)[nH]cc1[N+](=O)[O-] 97593,C#CCC(C(=O)NCC(C)CNC(c1ccn(CC(C)C)n1)=O)C1CC1 97594,C1(CNC(C2CCCC(OC)C2)=O)CC2(CCN(C(=O)C(CO)C(C)C)C2)CO1 97595,C1(C(=O)NCC2(C#C)CCCC2)CCC2(CC2)N1C(c1ccc(C)n1C)=O 97596,C1(CNC(c2cn(CCOC)c(=O)cc2)=O)CC12CCN(C(=O)C(C)C#N)CC2 97597,C1(C(N(CC(=O)OCC)C)=O)(CNC(=O)CN2CCCC2=O)CC12CCC2 97598,C(=O)(N=c1[nH]oc2c1COCC2)n1cc(C(=O)OC)c(O)nc1=O 97599,c1(C(C(=O)NCCCc2cncc(C(=O)OC)n2)(F)F)cc(Cl)nc(Cl)c1 97600,c1(C(=O)NC(C2CCN(C(c3ccc(Cl)nc3)=O)C2)C)cc2cc[nH]c(=O)c2s1 97601,C(C(CC)(CC)Sc1ccccc1)NC1C(CCC)COC1 97602,C(=O)(C(C)(C)C(N)=O)NCC1C(NC(C2N(C(=O)NC)CCC2)=O)CCCC1 97603,N1(C(C(C(=O)OCC)OC)=O)CCC(CC)CC1C(=O)NC(C)C(O)C(F)F 97604,C1(CNC(=O)C(N2CC=CCC2)=O)CCN(C2CCCC2)C1 97605,C(=O)(CC1CCNc2ccccc21)NC1(CO)CCCN(C(C2(C#C)CC2)=O)C1 97606,C1(N(C(CCOCCCNC(=O)NC)=O)C)CCC(C(F)F)CC1 97607,c1(C(=O)NCC2C(C)CN(C(=O)CS(N)(=O)=O)CC2)cnc2ncc(Cl)cn12 97608,CCC(CC(=O)N1CC(CC(C)(C)C)C1)C1CC1.n12cc(nn1)CCN(C)CC2 97609,N1(C(CCN(C)CC)=O)CCN(C(c2ccncc2C)=O)C2CC12 97610,N1(C(CC=CC(C)(C)C)=O)CCC=C(C(=O)NCc2ncccn2)C1 97611,C1(C)(NC(C2C(CCC)C2)=O)CCN(C(c2ncoc2-c2ccccc2C)=O)C1 97612,c1(-c2n(-c3c(C)cccc3)nc(CS(C)(=O)=O)n2)cc(C)c2[nH]nnc2c1 97613,C1(C(N2C(CCNC(C(N3CCNC3=O)C)=O)CCCC2)=O)CC2(CC2)CN1C 97614,Cc1ccc(SCC(=O)NCC2C3CN(C(C4CCCSC4)=O)CC23)cc1C 97615,c1(C(=O)N2C3CC3C2)c[nH]nc1C1CCC1.C1(C(=O)NN2CCCC2)CC1[N+](=O)[O-] 97616,N1(C(c2nc(CC)sc2)=O)CC2(CC2)CC1C(=O)NCC1(O)CCCOC1 97617,C1(C(=O)NC(C2CCN(C(c3cnco3)=O)C2)C)CCCC(=O)N1C 97618,Cc1cnc(F)cc1-c1cnccc1C(c1ccccc1)Nc1nccc(Cl)c1Br 97619,NC(=O)CCC(=O)NCC1CCCCN1C(C1(F)CCOCC1)=O 97620,CN1CCC(N(C)C(C2COCCC2NC(c2cncc(Cl)c2)=O)=O)CC1 97621,C(C(C)(C)C#CC(=O)NC(c1cccnc1)CO)NC(CCc1c(C)noc1)=O 97622,N1(C(C(C)SCC)=O)CC(CCNC(c2cn(CC)nc2C(C)C)=O)C2(CC2)C1 97623,N#Cc1ccc(NC(=O)C(=O)NC(C2CCCCC2)Cc2ccccn2)cc1F 97624,C(=O)(C#CC1CCC1)N1CCCC(N(C(c2ccc(N(C)C)nn2)=O)C)C1 97625,c1(C(N2CCCN(C(c3cccnc3)=O)CCC2)=O)cc(Br)c2occc2c1 97626,C1(NCc2cc(C)nn2-c2ccccc2)CC(N=c2[nH]cnc3cnccc23)C1 97627,C1(NC(c2c(C)c[nH]n2)=O)C(C)(C)CN(C(C2CCNC(=O)C2)=O)CC1(C)C 97628,C1(C)(CNC(CC(C)OC)=O)COCCN(C(c2csc(-c3ncc[nH]3)n2)=O)C1 97629,CC1(C)CC(C(F)F)CN1CC(C1CCOC1)F 97630,c1(OC)cc(CNC2(CC(N3CCCC(CO)C3)=O)CCC2)cc(Cl)c1 97631,C12(CNC(C(CCC(C)C)O)=O)CCCC(CN(C(=O)C=C3CCC3)C1)C2 97632,c1(C(N(c2ncc(F)cn2)C(C23CC(N)(C2)C3)=O)=O)cc(Cl)cnc1F 97633,c1(C(N2C(C)CC(CNC(=O)CC3CCC(=O)N3)C2)=O)cnc2c(c1)CCC2 97634,C1(C(N(CCCCNC(C(C2CC(F)(F)C2)OC)=O)C)=O)CCC2CC1CO2 97635,C12(CNC(CCC(=O)OC)=O)CCCC1CCN2C(c1ccsn1)=O 97636,N1(Cc2nc(CC)on2)CC(c2cccc(C(F)(F)F)c2)OC(C)C1.C1(=O)C(=O)CN1.OC 97637,c1(C(=O)NCC(CCNC(c2ccc(F)c(F)c2F)=O)O)cccc2c[nH]nc12 97638,c1(C(=O)NC(c2cn(C)nn2)C(=O)NCc2n(CCC)ncn2)ccc(Cl)cc1 97639,CCCC(C(=O)N1CC(CNC(C2CNC(=O)N2C)=O)C1)C(C)C 97640,c1(CCCC)cc(NCC2CN(C(C3CC4CCC3C4)=O)C2)n2ncnc2n1 97641,c1(C(N2CC(CNC(C(C(C)O)N(C)C)=O)C2)=O)ccc2c(n1)CCCN2 97642,N1(C(=O)COCC2CC2)CCC2CCN(C(=O)CCc3cscn3)CC2C1 97643,C(=O)(CC(C)C(C)(C)C)N1C(C(=O)NC2(C(=O)OC)CCCCC2)CC1C 97644,c1(C(C(=O)NCCC2CC2)N(C2CC(OC)C2)C)ccncc1 97645,c1(C(N2C(CNC(c3cn(CC(N)=O)nn3)=O)CCC2)=O)cc(N)cc(N)c1 97646,C12(CCNC(CCc3c(C)cccc3)=O)CCC1CN(C(=O)C(C)(C)CF)C2 97647,C1(CNC(=O)C=CC2CC2)CC2CCC1N2C(C1CC2CCC(C1)S2)=O 97648,CC1CCCC(C(=O)NC2CCCC2CN=c2[nH]nc(C3CC3)s2)CC1 97649,N1(C(c2cc3ccc(F)cc3[nH]2)=O)CCc2ccccc2C1CO 97650,c1(C(=O)NCC(CC=C)NC(c2ccc([N+](=O)[O-])[nH]2)=O)cccn2cc(C)nc12 97651,C#CC1C(C(=O)NC2CCC(CNC(c3cccc(N(C)C)c3)=O)CC2)C1(C)C 97652,C(=O)(CS(=O)(=O)CC(=O)NCC(CNC(c1ccnc(S)c1)=O)C(F)(F)F)OC 97653,C#CCCCC(=O)NC(C)CCN(C)C(c1ccncc1Cl)=O 97654,Cc1cn(C)nc1CNC(C1(NC(=O)CCCOC(=O)N(C)C)CCOCC1)=O 97655,C1(CNC(C)C)CN(c2ccnc(NCCC3CCCC(C)C3)n2)CCO1 97656,N1(CCNC(C2CCCCC2F)=O)CCCN(C(c2cc(CF)on2)=O)CC1 97657,C=C(Cl)CC(C(=O)NC(C)CCN1CCCC1)NC(c1cnc(Cl)s1)=O 97658,N1(C(C2(NC(N)=O)CC2)=O)CCS(=O)(=O)C(CCNC(c2cccnc2S)=O)C1 97659,C(=O)(C(C(C)NC(=O)CCCn1cccn1)C(C)C)NCc1cc(C)oc1 97660,c1(C(=O)NCCN(CC(C)O)C(C2CCOC2(C)C)=O)ccc(C(F)(F)F)cn1 97661,n1(CC)ccc(C(N2CCC2c2cn(-c3ncc(C)cn3)nn2)=O)c1C 97662,C1(NC(COCP(C)(C)=O)=O)CCC(NC(C2CCCCC2C(F)(F)F)=O)CC1 97663,C1(C(=O)NCC2(COC)CCCC2)C2CCC(C2)N1C(=O)CN(C1CCCC1)C 97664,c1(C(=O)NC(CN(C)C(C2CS(=O)(=O)C2)=O)CO)cc(C2CC2)ccc1F 97665,CCCC(CC)C(=O)NCc1cn(C2CN(C(=O)C(C)(C(C)C)OC)C2)nn1 97666,N1(C(C2C3(CCN(C(=O)CCN4CCCC4)C3)C2)=O)CCc2ncncc2C1 97667,C1(CCC(=O)NC2(CNC(Cc3c(C)ocn3)=O)CC2)CCC(C2OCCO2)O1 97668,CN1CCC(NCCN2CCN(CCOC(=O)CCC3CC3)CC2)CC1 97669,C1(CC#C)(C(=O)NCCC2CC(NC(=O)CNS(=O)(=O)NC)C2)CCCCO1 97670,C1(OC)CC(CNC(=O)CC2C(C)(C)C2(C)C)N(C(c2ccc(C3CC3)o2)=O)C1 97671,CC1COC2(CCN(C(=O)Nc3sc(I)cc3Br)CC2)O1 97672,N1(C(c2c(CCC)n(C)nc2)=O)CCC(C)(NC(C2CC2C(C)O)=O)CC1 97673,C1(CCNC(c2cc(COC)on2)=O)CN(C(=O)Cc2csc(C)c2)CCO1 97674,O=S(=O)(C(F)(F)F)NCC(C)NC(c1ccccc1)Cc1ccccc1 97675,CCC(CC(=O)NC1CN(C(=O)Cn2nc(C)oc2=O)CC1(C)C)C(F)F 97676,C1(CC(=O)NC2COC(C3CC3)C2)CC2(C1)CN(C(C13CCC(CC1F)C3)=O)C2 97677,N1(C(c2n(CC)nnc2)C(=O)NCc2ccccc2)CCC(N=[N+]=[N-])C1 97678,C1(C)(NC(c2ccc(CNC(C)=O)s2)=O)CCN(C(=O)CC2CCNC2=O)C1 97679,c1(CC(=O)NC(C)(C)CNC(C2COC(=O)O2)=O)ncn2c1CCC2 97680,N1(C(C2C(C(C)(C)C)C2)=O)CC2(CCCN(C(c3cccn3C3CC3)=O)C2)C1 97681,C(=O)(CC(C)(C)C(F)F)NC1CN(C(CNC(CC)=O)=O)CC1(C)C 97682,C1(C(C(=O)NCC=C=C)C)CCN(C(c2ccc(C3CC3)cc2)=O)CC1 97683,Cc1nn2ncccc2c1C(=O)NC1CC2C1CCN2C(=O)C(F)F 97684,N1(C(CNC(CC)=O)=O)CCC(CO)(NC(c2ccc(CC)[nH]2)=O)C1 97685,CC1CCC(N(C(=O)CCNC(=O)OC(C)(C)C)N2CCN(C)CC2)C1 97686,C(=O)(CCC(=O)NC1CCCC1)NC(CNC(CC(=C)Br)=O)C1CCC1 97687,C(=O)(C1=CCC(C(F)(F)F)OC1)NC1CCC(N(C(C(C(C)C)F)=O)C)CC1 97688,C(=O)(CCCC(=O)N1CC(NC(=O)CCC2OCCO2)CC(F)C1)NCC 97689,N1(C(c2ccc(NC(C)=O)s2)=O)CCCC(NC(=O)C2=COCCO2)CC1 97690,C1(CNC(C(=O)NC(C)C)=O)CC(CNC(C2(F)CCC2)=O)CO1 97691,c1(OC)ccc2ccc(C(=O)OCc3nc(Cl)ccc3F)cc2c1 97692,n1(CCOC)cc(C(=O)NCC(C2CCCC2)NC(=O)C2=CCCO2)c(C)n1 97693,Cc1cc2[nH]c(C(=O)NC3CN(C(C4CC4C(C)O)=O)CC3(C)C)cc2s1 97694,O=C1NCCN(C(=O)NC2CCN(Cc3ccccc3)CC2)C1CC(F)(F)F 97695,N1(C(=O)Cc2nc(Cl)cs2)CCC(F)(F)C(C(=O)NCc2ccccc2)C1 97696,C(=O)(N(CC1CCCCC1)OCCC(C)C)c1scc(C(=O)OC)c1 97697,C1(CNC(C2OCCN(C(CN(CC)CC)=O)C2)=O)CCC=CCCC1 97698,c1(CCNC(=O)Nc2ccc(N3CCOC3=O)cc2)ccc(-n2cnnc2)cc1 97699,CC(C)CC(CNC(=O)CN1CCCC1CO)NC(c1cn(C)nc1C(F)F)=O 97700,c1(OC)ccc(CNC(c2nc(CN(C)CC3CSC3)cs2)=O)c2cccnc12 97701,N1(C(C(C)OCC2CC2)=O)CC2CCC1C(CNC(C1C(C)OC(C)C1C)=O)C2 97702,C(C(C(=O)NC1(CNC(=O)C(O)C2CC2)CCCCCC1)C(C)(C)C)OCC=C 97703,CCCC(C)(C)CC(=O)NCC1CN(C(=O)CC2CC23CC3)CCN1C 97704,N1(C(CCC(C)C)=O)C2CCCC1CN(C(=O)CNc1ccccc1[N+](=O)[O-])C2 97705,C1(C(N(C)CCNC(=O)CNc2ccccc2Cl)=O)CC1C1CCCCC1 97706,C#Cc1cnc(C(N2CC(NC(C3CC(C)(C)CO3)=O)C3CCCC23)=O)c(C)c1 97707,N1(C(c2ccc(C#N)c(Cl)c2)=O)CCC2(CCN(C(C34CC(F)C3C4)=O)CC2)C1 97708,C1(C(=O)NCCN(OC)C)C2CCC(C2)N1C(=O)CC1CCC(=O)C1C 97709,C1(N(c2c(F)ccc(C)c2)C(=O)C(C)n2cnnn2)CCC12CCNCC2 97710,c1(OC)cc(Cl)ccc1C(=O)NCCCOCCNC(=O)C(C)SC 97711,Cc1c(NC(C2CCCN(Cc3c(Br)cncc3Br)C2)=O)ccc([N+](=O)[O-])c1C 97712,Cc1cc(F)ccc1-n1cc(C(=O)NC(c2cccnc2F)C)nn1 97713,C1(C(=O)NCc2c(C)nc(N(C)C)s2)C(C)CCCN1C(=O)CN1CCCC1 97714,c1(C(=O)NCCCN(C)C(c2nc(O)nc(O)c2F)=O)nnn2c1C(=O)NCC2 97715,Cc1ccc(Cl)cc1C(=O)NC1CN(C(=O)COC2CCN(C)CC2)CC1C 97716,CCC1=C(C(=O)N2CC(COC)C2)SCCO1.C(=O)(C(F)(F)c1cnn(C)c1)N 97717,N1(C(C(CCCC)O)=O)CCC2(CCC(CNC(c3ncoc3C)=O)OC2)CC1 97718,C(=O)(C1=CC2(CCOCC2)C1)NCC(C)CNC(C1COc2ccccc2O1)=O 97719,CCCCC(O)CC(=O)NC(C)(CC)CCNC(c1cc(OC)nc(C)c1)=O 97720,C(=O)(C(F)CC(C)(C)NC(=O)C(CCSC)OC)NCC(C(CC)C)CO 97721,C(C)(C(=O)NN1C(=O)CCC1c1cccs1)(OCC)OC 97722,C1(NC(c2c[nH]nc2F)=O)CC2(C1)CC(NC(=O)C(O)C1CCCC1)C2 97723,CC1CCC=C1C(=O)N(C1CCN(C(=O)CCc2ccc(F)nc2)CC1)C 97724,CC1CCN(C(C2CC(N=[N+]=[N-])C2)=O)C1CNC(=O)CCS(C)=O 97725,c1(CNCCCC2(NC(C3(c4c(C)cno4)CC3)=O)CC2)c(C)nn(C)c1C 97726,c1(C(=O)NCC(C2CCCCC2)NC(C(CCOC)C)=O)ccc(C)nc1C 97727,n1(CC)cc(C(=O)NCC2CN(C(=O)CCC3CCC(=O)N3)C2)nn1 97728,CC(C)C(C(=O)N1CC(CC(C)(C)CNC(c2coc(CO)c2)=O)C1)n1cnnn1 97729,c1(C(N2CC(NC(c3cc(C(C)C)[nH]n3)=O)(CO)C2)=O)ccc(Cl)c(Cl)c1 97730,C1(C(=O)NCCCCCC)CN(C(=O)CC(C)(C)C(F)F)CCC1(C)C 97731,c1(C(=O)OCC#N)ccc(C(=O)NCC2CCCN(C(=O)C=CCO)C2)cc1 97732,N1(C(CCSc2ccc(C)cc2C)=O)CC2CCN(C(=O)C(O)C(C)C)CC2C1 97733,Cn1c(Cn2ccnc2-c2cnc(Cc3ccccc3)nc2)nc2ccccc12 97734,C1(CC)(CC)CC(NC(C2(C)CCOC2)=O)CN1C(c1ccc(SC)o1)=O 97735,c1(CC(N2C(CNC(=O)CC3CC3)CC(O)C2)=O)c[nH]c2cccnc12 97736,N1(C(c2cn(C(C)C)nn2)C(=O)NC2CCCC2)CCCC(C)(C#N)C1 97737,C(CC(=O)N1CC=C(CCNC(=O)C(C)(C)C)CC1)(C(F)(F)F)OC 97738,CC(O)(C(=O)N1CC2(NC(=O)C=CCOCc3ccccc3)CC1C2)C(F)(F)F 97739,C(=O)(C(CC(F)F)NC(C1CC1C(=O)OC)=O)NCCOCC 97740,C1(CNC(=O)COCC2CCCO2)CN(C(c2cnn3c2OCC3)=O)CC12CC2 97741,C(CN=c1[nH]ccnc1F)C1CCC(NC(c2nc(CC)sc2)=O)C1 97742,Cc1ccc(C(C(=O)N(C2CC2)CC2CC2)N2CCC2C(=O)OC(C)(C)C)cc1 97743,N1(C(C(C)Nc2cccs2)=O)CCCC1c1nc(C(=O)NC2(C)CC2(F)F)cs1 97744,c1(OC)ccc(C(=O)Nc2nc(C(=O)Nc3ccccc3N(C)C)cs2)c(Cl)n1 97745,N1(C(CCC(=C)C)=O)CC2(CC(NC(C3CC(O)CN3C(N)=O)=O)CO2)C1 97746,C(C(C)(CN(C)C(c1cccc(C(F)(F)F)c1)=O)CO)OC 97747,C(CC1=CCN(C(=O)Cc2cnccn2)CC1)NC(CN(C)C1CC1)=O 97748,C1(N(C(C(C)Sc2ncccn2)=O)C)CC2CCC(C1)N2c1ncc(Cl)c(O)n1 97749,C1(NC(c2c(C)con2)=O)CC2CCC(C1F)N2C(C1CCCC(C2CC2)O1)=O 97750,C(=O)(C(C(C)(C)C)N(C)C)NCCSCC(=O)N(C1CN(C)CC1O)C 97751,N1(C(COC(C)C)=O)CCC2CCN(C(c3nc(=O)n(C)[nH]3)=O)C2C1 97752,C(c1c(Cl)cccc1Cl)=CC(N1CCN(C(C2CC2F)=O)C(CO)C1)=O 97753,N1(C(C(C(C)C)CO)=O)CCc2c(CNC(=O)CSC(=N)N)cccc2C1 97754,c1(C(C)=O)c(NCCCCC(C)NC(=O)C(c2ccc(C)s2)C)ncnc1Cl 97755,c1(C(N(CC(N2CC(CC3CC3)C2)=O)C)=O)ccnn1C(F)F 97756,c1(C(=O)NCC(C)NC(C(C2CC(F)(F)C2)OC)=O)cnc2c(c1)NCC(=O)N2 97757,c1(OCC)c(C(=O)NC2CCN(C(C3(C(F)F)CC(F)(F)C3)=O)C2)cccc1F 97758,C12(C(=O)NCCCC(C)(C)NC(CC(CC)C)=O)CCC(=O)N1CCS2 97759,CN1CCc2cc(CC(=O)NC3(CNC(c4nccn4C)=O)CCOC3)ccc21 97760,Cc1ccc(C(N2CC(NC(=O)Cc3n[nH]cc3Br)C(C)(C)C2)=O)cc1C#N 97761,C1(CC(=O)NCC23C(CN(C(Cc4ccc(C)cc4)=O)C2)C3)CCOCC1(C)C 97762,C12(NC(c3n(CC)ccn3)=O)CCC1CN(C(=O)C(C1CC1)N(C)C)C2 97763,C1(C(C)C)N(C(=O)Nc2nc(N3CCOCC3)ncc2Cl)CC12CCS(=O)(=O)CC2 97764,c1(CCC(=O)N(CCCNC(C2OCCCO2)=O)C)ccc(Cl)nc1 97765,C(=O)(CC(F)(F)CC)N(CC(=O)NC(CCSCC)C)C 97766,c1(C(=O)NCC2CCN(Cc3cnc(CCC)s3)CC2)cc(Br)cnc1O 97767,c1(C(C(=O)Nc2cnn(C(C)(C)C)c2)C)cncnc1.C(=O)(CN1C(=O)C1)OC 97768,C1(C(=O)NCCOCCC2CC2)(CNC(c2c[nH]c(=S)cn2)=O)CC2(CC2)C1 97769,c1(C(=O)NC2C(CN(C(C(CCOC)OC)=O)C)CCC2)cnc(O)cc1OC 97770,C(=O)(CCCC(C)(C)C)N1CC(C)C(CNC(C2C3CC4C(C3)C24)=O)C1 97771,N1(C(C2C(C)OCCC2)=O)CC2CCC1C(CNC(=O)CC(C)(C)C)C2 97772,Cc1ccccc1-c1cnc(CNC(=O)NCCN2CCSCC2)o1 97773,c1(C(=O)NC(C(C)NC(c2cc(C)ns2)=O)CO)ccccc1SCC#N 97774,C1(CNC(C2(C)CC=CCO2)=O)CC2(CCC2)CN1C(=O)COc1cccnc1 97775,CC1(NC(=O)Cn2cc(Br)cn2)CC(NC(C2(CC3CCC3)CC2)=O)C1 97776,N1(C(c2ccc(CC)[nH]2)=O)CCC(N(C(=O)C(C)COCC)CCO)CC1 97777,Cc1cc(Cl)c(Cl)cc1C(N1CCC(C)CC1C(=O)OC(C)(C)C)=O 97778,c1(C(=O)NC(CC)CN(C(=O)Cc2cc(C)[nH]n2)C)cccn(C(C)(C)C)c1=O 97779,N1(C(CCC#CC)=O)CCc2ccccc2C1CNC(=O)CCN(C)C(C)=O 97780,N1(C(CN(CCOC)C)=O)CCCC(C(C)C(N2CC(CO)CC2CO)=O)C1 97781,c1(C(N2CCC(C(C(=O)NC3CC(C)(C(=O)OC)C3)F)C2)=O)ccc(C)nn1 97782,C1(C(N2CCC(CNC(C3(CC(C)C)CCC3)=O)C2)=O)C2CCCCC12 97783,C1(CC)C(C(N2CC(F)(CO)C2)=O)CCN1C(c1cc(C)n(C)n1)=O 97784,C1(CNC(CCOCCN(C)C)=O)(NC(C2(CO)CCOC2)=O)CCCC1 97785,C(=O)(C(CC)C(F)(F)F)NC1CC(CCNC(C2(CC=C)CC2)=O)C1 97786,CCC(CC(F)F)C(=O)N1CCC(C2(NC(c3cccn4ccnc34)=O)CC2)C1 97787,c1(CC)cc(C(=O)NC2C=CC(CNC(=O)C(C)=C3CCC3)C2)ccn1 97788,c1(C(N(CCCNC(C2CCCC23CC3)=O)CC)=O)ccc(F)c(CO)c1 97789,Cc1coc(C)c1C(=O)NCC1CCN1C(C1(c2ccc(Cl)cc2)CCCCC1)=O 97790,c1(C(=O)NC(CC(=C)C)C(=O)NC(C)CCCO)cccc2[nH]ncc12 97791,C1(NCCOC)Cc2ccc(C)cc2S1.c12cccnc1C(=O)N(C)CCNC2=O 97792,Cc1cncc(CCNC(C2(NC(=O)C=CC3CCOC3)CSC2)=O)n1 97793,c1(NCCOC)ccc(C(=O)NC2CCCCC2NC(c2cocc2C)=O)cc1 97794,c1(C(=O)Nc2cncc(C(=O)NCc3c(C)cccn3)c2)ccc2c[nH]nc2c1 97795,N1(C(C(COC)(C)OC)=O)CC2CC(NC(c3c(Br)nnn3C)=O)C1C2 97796,c1(NC(c2n(CCC(=O)OCC)nnn2)c2ccns2)cc(OC)ccc1C 97797,C=CCC(CNC(C1CCCC(C#N)C1)=O)C(=O)N1CCC(C)(CO)C1 97798,Nc1cncc(C(N2CC(CO)(NC(C3CC3c3cn[nH]c3)=O)C2)=O)c1 97799,C1(NC(C(c2ccccc2)C)=O)CCN(Cc2c(O)cccc2F)CC1O 97800,C(=O)(CC(C)C(=O)N(C1CCC(NC(c2nccn2C(C)C)=O)CC1)C)OC 97801,CCCCC(C(=O)N1C2CCCC1CN(C(C1(C3CCCO3)CC1)=O)C2)C(C)C 97802,C1(C(=O)NCC(C(C)O)O)CCN(C(=O)C2=CCCC2)CCO1 97803,C(=O)(CCC(C)(C)NC(=O)CNC(C1CC1C)=O)NC(C(CC)(C)C)C 97804,C=C1CC(C(F)(F)F)(C(=O)N(C)CC2CCN(C(=O)C(C)OCCOCC)C2)C1 97805,CCC(CNC(C1(c2cc[nH]n2)CC1)=O)(CC)NC(=O)C(C)OCC(F)(F)F 97806,C#CC1CCC(C(N2CCCC(N(C(=O)CCOCC(F)(F)F)C)C2)=O)CC1 97807,C1(NC(c2cc(C)n(C)n2)=O)CC2CC(NC(c3ccncc3O)=O)CC2C1 97808,N1(C(C(CCC)=CC)=O)CCC2CN(C(=O)C(CC#N)c3ccccc3)CC2C1 97809,CC(C(=O)NCCC(O)CNC(c1ccc(C(F)F)c(Cl)c1)=O)P(C)(C)=O 97810,C1(C(C)C)CC(NC(=O)C(N)Cc2cccc(Cl)c2)CN1C 97811,CC1CCCC1(C)C(=O)NCc1cccc(CN(C(=O)Cn2cnc(=N)[nH]2)C)c1 97812,c1(C(=O)NC2CC3CC(NC(=O)CN4CCCC4=O)C3C2)occ2c1CCOC2 97813,CC1CN(C)CCN1C(=O)CC1CCCN1C(c1ccc(F)cc1I)=O 97814,c1(CC(=O)NC(C(C)NC(c2ccccc2Cl)=O)CO)ccc2c(c1)COC2 97815,c1(OC)cc(CN2CCCC2C(N2CCOC(C(N)=O)C2)=O)c(F)cn1 97816,O=c1[nH]ccn2c(CN=c3[nH]c(Cl)ncc3Cl)cnc12 97817,C1(CCCCC)CC1C1CC1C(=O)N(C(c1c(C)noc1CCC)=O)CC 97818,n1(CC(=O)NCC2CN(C(C(COC)NC(C)=O)=O)CC2O)nc(O)ccc1=O 97819,C1(CNC(Cn2c(C(C)C)nnn2)=O)CCCCN(C(=O)C(C)CC2CC2)C1 97820,CN1CCOC(CNC2CCC(CNC(c3cnccc3Cl)=O)CC2)C1 97821,C1(NC(C(C=C)OC)=O)CC=CCC1C(=O)NC1CC2C=CC1C2 97822,c1(C(=O)NC(C)CNC(c2c[nH]c(Br)c2)=O)ccc(F)cc1OC(F)F 97823,Cc1c(C(=O)NCC(C)(Cn2cccn2)NC(=O)C(O)C(F)F)cccc1CO 97824,Cc1ccc(C(=O)NCCn2ccc(C(=O)N(C3COCC3(C)C)C)c2)n1C 97825,C1(c2cccnc2)(C(=O)NCC(CCNC(c2c(C)scn2)=O)O)CC(F)(F)C1 97826,c1(OC)cnc(Cl)[nH]c1=NC1CC2CN(C(=O)CCc3ccc(F)nc3)CC12 97827,Cc1cnc2n1C(C(=O)N1CCC(C)(NC(c3csnc3Cl)=O)CC1)CCC2 97828,C#CCC(C)(C)C(=O)NCC(CNC(c1ccnn1C1CCCC1)=O)C(F)(F)F 97829,S(=O)(=O)(c1cccc(Cl)c1)NCC(=O)NCC12N(C(CCC=C)=O)CC(CC1)C2 97830,C12(NC(C(CC)C(C)C)=O)CCCN(NC(=O)OC(C)(C)C)CC1C2 97831,C1(NC(c2[nH]cc(CC)n2)=O)CC2CC1N(C(=O)Cc1cccc(C)c1Cl)C2 97832,N1(C(C(C)SC)=O)CC(C2CN(C(=O)COc3ccsc3)C2)C1 97833,N1(C(c2cc(OC)cc(C)n2)=O)CC2CC(C)N(C(=O)CC3CNC(=O)C3)C2C1 97834,O(NC(=O)CCN(C(=O)CC1CCC(C#N)C1)CCO)CCCC 97835,C1(CCC)CN(C(=O)C(C)C=Cc2ccccc2)CCN1C(=O)CC 97836,N1(C(c2c(CC(C)C)onc2)=O)CC(NC(c2cn(CCO)nn2)=O)CC(O)C1 97837,Cc1cc(Cl)ccc1NC(=O)C(C)(C1CCC1)NC(C1CC(CF)C1)=O 97838,N1(C(c2c(C)c(Br)no2)=O)CCC(C)(NC(C2CC(CF)C2)=O)CC1 97839,c1(C(C(=O)NC2CCOC2)N(CC(C)C)Cc2cccnc2)nc(C2CC2)cs1 97840,N1(C(C(F)=CC)=O)CCN(C(c2cnc3n2CCS3)=O)C(CS(C)(=O)=O)C1 97841,N1(C(Cc2cn(CC)nn2)=O)C(CNC(=O)COC(C)=O)CC2COCC12 97842,N1(C(C2CCCC(C)(C)C2)=O)CCC2(CCCCC2NC(=O)Cc2cn[nH]c2)C1 97843,Cc1nn(C)c(C(=O)NCC2(C)CC(NC(=O)Cn3cc(C(F)F)cn3)C2)c1Cl 97844,c1(C(=O)NCC(CCOC)NC(C2CN(C(C)=O)C2)=O)cc2cc(Cl)ccc2o1 97845,c1(C(N2C(C(N3CC(C#C)C(O)C3)=O)COCC2)=O)cccc2c[nH]nc12 97846,C(=O)(C1CCc2c[nH]nc21)NCCC(C(C)C)NC(COCCOCC)=O 97847,C(=O)(C(C)C(C)C)NC(C(C)NC(c1n(CC)ncn1)=O)CO 97848,C(CCC(C)(C)C(=O)NCC(O)CC(C)C)NC(C(C)=CC(C)(C)C)=O 97849,CCCCCCCCC(=O)NC(CC)CCCC(=O)NCC12CCC(CC1O)C2 97850,C1(CNC(CC(C=C)C)=O)CC2CCC1N2C(c1ccc(CO)s1)=O 97851,Cc1cccc(Cl)c1C(N1CCC(C)C1CNC(=O)CCOCCN(C)C)=O 97852,C(=O)(C#CC1CCCCC1)N(C)CC1CCCCN1C(C1CC(O)CN1C)=O 97853,CCC(C)C(C(=O)NCCCCNC(=O)CC(F)(F)F)NC(N)=O 97854,C1(C(=O)NC2CCCC2)CCCN1C1CC1.C12(CC1)N(C)C2=O 97855,n1(CC(=O)NCC2(F)CC(NC(Cc3cn(CC)nc3)=O)C2)nc(O)ccc1=O 97856,C1(C(N2CC(O)(C(C)NC(Cc3cc(C)sc3)=O)C2)=O)CCCCN1N=O 97857,c1(C(=O)NCC(C2N(C(C(COCC)C)=O)CCC2)(C)C)c(OC)cccc1Cl 97858,c1(NC(C(=O)Nc2cn(CC#C)nc2)=O)ccc(C(OC)OC)cc1 97859,CCCCCC(=O)NC(Cc1ccco1)C(=O)NCc1cc(C(N)=O)no1 97860,c1(OC)cc(N)c(Cl)cc1C(=O)NC1(C)CC(NC(=O)C(C)CC2CCCC2)C1 97861,C=C1CON(C(=O)C23CC2CCN3C(=O)Cc2cccnc2O)C1 97862,C(N=c1nc2sccc2c(N(C2CCCCCCCC2)C2CCN2C2=CC=C2CO)[nH]1)C1(C)CC1(Cl)Cl 97863,N1(C(C=CC(=O)OCC)=O)CCC(NC(=O)C=CCOC)C1Cc1ccncc1 97864,CCS(=O)(=O)CC(C)N=c1[nH]c(=NC(C)c2ccccc2Br)[nH]c2ncn(C)c12 97865,CON(CCC(=O)NCC1CCCCN1C)C(=O)C1CCCC(=O)N1C 97866,C(CC(F)(F)Cl)COC(C(C1(CCO)CC1)NC(=O)OC(C)(C)C)=O 97867,C1(NC(C=C(C)C2CC2)=O)CC(CNC(c2cc(CO)c(C)o2)=O)C1(C)C 97868,N1(C(CC=C=C)=O)CC2CC(NC(=O)CS(=O)(=O)CCC)C(C2)C1 97869,CCCC(C(O)C(=O)NCCC1CCC(C)(C)C1)NC(c1cc(C)nnc1C)=O 97870,CCC(C)(C(=O)NCC1(C)CC(F)(F)CN1C(c1ccc(F)cc1)=O)C(N)=O 97871,C12(C(N3CC(O)(CNC(CSc4ccc(C)cc4)=O)C3)=O)CCC(C)(CC1)OC2 97872,N1(C(C2C(CC)CCCC2)=O)CCCC(C2CN(C(=O)C(F)(F)C(C)O)C2)C1 97873,O=C(CCC(=O)N1CC=CC(NC(=O)CC2CCCCC2)C1)c1cccc(Cl)c1 97874,c1(COC(c2ccc(-c3ccc(OC)nc3)nc2)=O)ccc(OC)cc1F 97875,C(=O)(CC(CC)C(F)F)N(CC(=O)NCc1cccnc1)CCC 97876,N1(C(C(CC2CC2)OC)=O)CC2(CNC(c3scnc3C3CC3)=O)CCC1CC2 97877,C1(C(=O)NCC(C)(C2CC2)NC(c2cnc(COC)s2)=O)CN2CCN1CC2 97878,c1(C(C(=O)NCC2N(C(c3cc(CO)sn3)=O)CC2)(F)F)cc(Cl)ccc1Cl 97879,C1(NC(C2N(CCC)CCC2)=O)CCCN(C(C2(CC)COC2)=O)C1 97880,c1(SC(c2n(CC(=O)N(C)C)nc(-c3cccnc3)n2)=O)cccc(Cl)c1 97881,Cc1cc(CNC(C2(NC(c3cocn3)=O)CCSC2)=O)cnc1C 97882,CCS(=O)(=O)CC(=O)NCC12CCC(CN1C(=O)CC1CC(F)(F)C1)C2 97883,C1(C(=O)NC(C(=O)N(CC)CC)C)CN(C(=O)Cc2scnc2C)CC1C1CC1 97884,C(=O)(CC(C)(C)C#N)NCC1CN(C(c2ccc(CCCC=C)cc2)=O)CC1C 97885,c1(-n2c(C(C3(C(C)C)CC3)NCCCc3cccs3)nnn2)ccc(F)cc1 97886,Cc1ncc(C(N2CC(NC(=O)C3=NOCC3)C(c3ccccc3)C2)=O)n1C 97887,N1(C(C2(CC=C)CN(C(=O)CC(C)CC(=O)OC)C2)=O)CC(C)(C)CCC1C 97888,C1(C2CCC2)(C(=O)NCCCC(C)NC(C2CCC=CO2)=O)CCC1 97889,CC(C)CC(C(=O)N1CCCC1CN1CCC(CNC(=O)CCF)CC1)N(C)C 97890,C1(COC(C)C(N2CC(C)(OCC(=O)NC3(C)CC3C)C2)=O)CCCCO1 97891,C(=O)(CCCCC(=O)NCC1CCN1C(C1(O)CC1)=O)NC 97892,C1(C(=O)ONC(C2CCN(CC#C)CC2)=O)CN(C(=O)CSC(F)F)C2CCCCC12 97893,c1(C(N2C(CNC(C(C=C)OC)=O)CCC2)=O)cc(C)cc(O)n1 97894,c1(NC(C(c2ccc(SC)cc2)N(C(COC)C)C)=O)ccc(F)cc1 97895,c1(C(=O)NCC=CC)n[nH]cc1CNC(=O)C(C)n1cccn1 97896,c1(C(C)CC(=O)NC2(CO)CN(C(=O)CCN3CCCC3)C2)cccc(F)c1 97897,CC1CNC(=O)CN1C(C1(NC(C2(C3CCCCO3)CC2)=O)CC(CO)C1)=O 97898,c1(CC(=O)NCC(CC)(C)NC(=O)C(C)CC(N)=O)sc2ccccc2c1C 97899,c1(CC(=O)Nc2ncc(-c3ccc(OCCCC)cc3)s2)cc(F)cc(Cl)c1 97900,CC1(C)CC(C(=O)Nc2cnc(F)nc2)(CNC(C2C(C)(C)C2(F)F)=O)C1 97901,N1(C(C=CC(C)NC(C(C)(C)NC(C)=O)=O)=O)CCC(O)(CO)C1 97902,N1(C(CCNC(C(C)(C)C)=O)=O)CCCC(O)(CNC(=O)CSCC(F)(F)F)CC1 97903,C1(C(N2CC(N(C(=O)CC3CC(F)(F)C3)C)C3(C2)CC3)=O)OCCOC12CCC2 97904,c1(CC(=O)NCC(C2CCCC2)NC(CC=C)=O)ccc(Br)cc1 97905,C1(CC)(NC(=O)CCCc2cccs2)CCN(C(=O)C(C)COC)C1 97906,N1(c2nnn(C)n2)CCCCC1CNC(C1COC(=O)N1C)=O 97907,Cc1ccc(C(=O)NCC2CN(C)CCN2C(c2ccccc2)=O)cc1[N+](=O)[O-] 97908,Cc1cc(CNC(=O)C(Cc2ccccc2Br)NC(C2CC2(F)Cl)=O)cc(O)c1 97909,c1(C(N(C(C)CNC(=O)Cc2ccc(OC(C)C)cc2)CC)=O)cn(C)c(O)n1 97910,C1(C(=O)NCC2C(C(F)(F)F)CN(C(CC=C=C)=O)C2)Cc2nnc(C)n2C1 97911,C1(C(=O)NCC(C(=O)OC)O)CCCCN(C(C2(O)CCOCC2)=O)C1 97912,N1(Cc2ccc(CC)cn2)CCC(F)(F)C(CNC(c2cnc3n2CCS3)=O)C1 97913,n1(CC(=O)NCC(CNC(C(CC)c2cccnc2)=O)F)c([N+](=O)[O-])cnc1C 97914,c1(OC)cccc(CC(N2CC3CC2C3C(=O)NCc2cccc(F)n2)=O)c1 97915,C1(c2nc(C)[nH]n2)COCCN1C(c1ccc(Br)cn1)C(=O)NCC(C)C 97916,Cc1ccc(F)c(C(=O)NC(Cc2cn[nH]c2)C(=O)NC2CC3CCC2O3)n1 97917,c1(C(=O)OC)ccc(C(=O)NC2CC2NC(c2cc(O)ccc2Cl)=O)cc1F 97918,C1(CC(C)C)CCN(C(=O)C(CCC2CCC2)NC(=O)COCC2CCOC2)CC1 97919,n1(CC(=O)NCCCOCCNC(=O)Cc2cc[nH]n2)cc(CO)nn1 97920,C1(NC(c2c(C)nc(C)o2)=O)CCC(C)N(C(C2CCN2C)=O)C1 97921,CCCCCC(C(=O)N(CC(C)(C)CNC(=O)COCCOCC)C)C(C)C 97922,c1(C2(F)CC(C(N3CCC(OCCNC(C(C)C)=O)C3)=O)C2)cccc(F)c1 97923,O=C(C1=CSCCO1)NCC1(CNC(c2ccc([N+](=O)[O-])o2)=O)CC1 97924,N1(C(CC2(OC)CCC2)=O)CCCCC1C(=O)N(C1CCC1C)C1CC1 97925,CCC(C(=O)N(CCCNC(=O)CC1CC(F)C1)C)NC(N)=O 97926,N1(C(CCCN(C)C)=O)CC2CCCC(C1)C2C(=O)Nc1n[nH]c(C(F)(F)F)n1 97927,C1(CC)C(=O)NCCN1C(=O)C(F)C(C)CNC(=O)COc1cnn(C)c1 97928,c1(CN(C2CC2)Cc2nc(C3C(C)N(C)CC3)on2)c[nH]c2cccnc2c1=O 97929,C(=O)(C1=NOC2COCC12)NC1CCC(C(N(C(C)C(C)(C)C)C)=O)C1 97930,N1(C(CC=CCCCCC)=O)CCC(C)(C(=O)N(C2CC3(CCC3)C2)C)C1 97931,c1(C(=O)NCc2c(C(N3C(COC)CCC3)=O)c[nH]n2)cncc(C)c1 97932,N1(C(C2N(C)CCC2)=O)CC(NC(=O)CCCC(C)(C)C)CC12CCCCC2 97933,N1(C(C2CCN(C)C2=O)=O)CC(C2CCN(C(c3ncn4c3CCC4)=O)CC2)C1 97934,Cc1cccc(C2(C(=O)NC(C3CCN(C(C4(O)CCSC4)=O)C3)C)CC2)c1 97935,C1(CC)CN(C(=O)CCOCC(C)(C)C)CCN1C(c1cnn(C)c1OC)=O 97936,CN1CCC2C(CCCN2C(c2ccc(Br)c(F)c2F)C(=O)NC2COC2)C1 97937,Cc1noc(C2CN(C(=O)CC(C)N(C(=O)C(C)OCCN(C)C)C)C2)n1 97938,Cc1cc[nH]c(=N)c1C(=O)NCC1(C)CCN(C(c2c(C)cnn2C)=O)CC1 97939,C1(NC(C2CC(=C)C2)=O)CC2CC(NC(=O)C(C)CC3CCCCC3)CC2C1 97940,C1(C(N(C2CCN(C(c3n[nH]c(O)n3)=O)C2)CCO)=O)CCC2CC2C1 97941,C(=O)(CCS(=O)(=O)c1ccc(F)cc1)N1CCN(C(CC=CC)=O)C(C2CC2)C1 97942,c1(C(N2C(C)(CC(=O)OCC)CC2)=O)cncc(-c2cc[nH]n2)c1 97943,N1(C(c2c(CC(C=O)(C)C)cnnn2)=O)CCN(C)C(COC)C1.CCO 97944,c1(OC)cccc(C(F)F)c1C(N1CCC(NC(=O)C(C)(C)CF)C(CO)C1)=O 97945,n1(CC)nccc1C(=O)NCC1CC1CNC(=O)CNC(c1cnn(C)c1)=O 97946,c1(C(N(C)CCNC(=O)C(c2cnn(C3CCCC3)c2)=O)=O)cccc(O)n1 97947,C=C=CC(C)C(=O)NCC(C)(C)OCC(=O)Nc1ccc(O)nc1 97948,CN1CCC2(CCN(C(C3C4CCC(C4)N3C(=O)CCC(F)(F)F)=O)CC2)CC1 97949,CC(C)C(O)C(=O)N1CC(CNC(=O)C(C)(C)n2cccn2)C1 97950,C1(C(N2CCC(N(C(=O)C(F)C3CCC3)CC3CC3)C2)=O)CC2(CCO1)CC2 97951,n1(CC)nc(C(=O)NCC2CCN(C3CCN(c4ccccc4)C3=O)C2)c(C)n1 97952,c1(CC)cnc(C(N2CC(NC(c3ccc(OC(C)C)cn3)=O)CC2C)=O)cn1 97953,c1(CNC(C(=O)NCCCCC)=O)ccccc1NC(C12COC(CN)(C1)C2)=O 97954,CC(C)C(C(C)C)NC(=O)NCC1CCC(C)C1 97955,C1(NC(C2C(NCC)C2)=O)CCN(C(=O)COCC(C)C)C1 97956,c1(C(N2CCC(N(C(=O)C(O)C(C)OC)CC)CC2)=O)cnn2c(C)ccnc12 97957,C1(C)(C(=O)NC(c2cccnc2O)C)C=CCN1C(c1cc(C2CC2)[nH]n1)=O 97958,C(=O)(CCC(N)=O)N(C1CCN(C(=O)C(CCSC)N(C)C)C1)CCC 97959,c1(C(=O)NC(C2CCN(C(=O)CSc3ccccc3)C2)C)ccc2scnc2c1 97960,c1(C(=O)OC)ccc2cnn(CC(=O)NCCN(C)C)c(=O)c2c1 97961,CC1CC=CCC1C(=O)NC(c1cnn(C)c1)C(=O)NC1CCC(F)CC1 97962,N1(C(C(CC)C)=O)CCCC12CCN(C(c1ccccc1[N+](=O)[O-])=O)C2 97963,N#CC1(C(N2CC3(C2)CN(C(=O)COCCN(C)C)C3)=O)CC2CC2C1 97964,c1(C(CCC)NC(N2CCC(c3cnc(C)s3)C2)=O)ccc(F)cc1 97965,N1(C(C=C)=O)CCC2(CCC2)C(NC(C2CCc3cncn3C2)=O)C1 97966,Cc1noc(C(=O)NC(c2ccc(CNC(=O)Cc3cnsc3)cc2)C)c1C 97967,c1(C(N2C(CC(N3CC(OC(=O)NC)C3)=O)CCC2)=O)ccc(Cl)cc1 97968,N1(C(C(C)O)=O)CCc2nc[nH]c2C12CCN(C(=O)C(F)Cl)C2 97969,C=CCC(Cc1ccccc1)N=c1nc2c(ncn2C)c(NC2C=CCCC2)[nH]1 97970,C1(CNC(C2C3C4CCC(C4)C23)=O)CCCC2CN(C(=O)CC3(O)CCC3)CC12 97971,N1(C(C2(CC#C)CCOC2)=O)CC(C)N(C(=O)CC2CC(C)(C)C2)C(C)C1 97972,c1(C(=O)NC(C)Cn2cc(CCCC(C)O)nn2)ccc2nccn2c1 97973,N1(C(C=Cc2ccc(C)o2)=O)CCOCC(CNC(c2c(C)nsc2C)=O)C1 97974,N1(C(C2(CC=C)CC=CC2)=O)CCN(CC(=O)NC(c2nn(C)cc2O)C)CC1 97975,CC(C)(C(=O)NCC(C1CCCC1)NC(=O)Cc1cnc[nH]1)Oc1ccccc1 97976,C12(C(=O)NC3C(CNC(C(C)OCCCC)=O)C3)CC3CC1C2C3O 97977,C1(C2CCOCC2)(C(N2CC(CNC(=O)CCc3ccccn3)C2)=O)CC1(F)F 97978,S(=O)(=O)(c1cc([N+](=O)[O-])ccc1C(=O)O)Nc1c(SC)cc(Cl)cc1 97979,c1(CC(=O)Nc2c(OC(C)C)cccc2)csc2nc(-c3cccs3)cn12 97980,C1(C(=O)NC(c2cccnc2O)C)CCCC(NC(=O)CCOC2CCC2)CC1 97981,C1(NC(c2nc(Cl)sc2Cl)=O)CCCCN(C(C2CN3CCC2CC3)=O)CC1 97982,N1(C(c2nc(COC)sc2)=O)CC2CC1C2CNC(c1n[nH]cc1F)=O 97983,Cc1ccc(F)c(CC(=O)NCC2(C)CCCN2C(=O)CC2CCCN(C)C2)c1 97984,c1(NC(C2CCN(C(C=C(C)c3ccco3)=O)CC2)=O)c(O)cccc1O 97985,c1(OCC)cccc(CC(N2CCC(CCNC(C3(C)CC(O)CN3)=O)C2)=O)c1 97986,c1(OC)c(C(=O)NCC(C)(C)CNC(=O)CCCc2ncc(C)o2)cccc1F 97987,n1(CC)cnc2c(NC3CC(NC(=O)COCC4CC4)C3)ncnc12 97988,C1(C2(C(=O)N(C)C)CCC2)CN(C2C(c3ccc(C)cc3)C2)CC1(C)C 97989,C1(C(C)C)CN(C(=O)CC(F)(F)F)CCN1C(=O)C(=O)NCC(F)(F)F 97990,c1(C(C(=O)NC(CC)(C)CNC(c2n[nH]cc2Br)=O)C)ccc(F)c(F)c1 97991,c1(C(=O)NCCN(C(C(C)OC2CCCC2)=O)CC(C)O)ccc(=O)n(C)n1 97992,C1(C(=O)Nc2cccc(CN3CC(C)OCC3)c2)Cc2c[nH]nc2CN1 97993,Cc1cc(C2CCCN2C(=O)NC(c2cccc(Cl)c2)(C)C)c(C)o1 97994,c1(C(=O)NCCC(CC)(CC)NC(=O)C(F)=C2CCC2)nn2cccnc2c1Cl 97995,N1(C2CCC(NC(C3(C(N)=O)CC3)=O)C2)CCN(C(=O)C=Cc2cnc[nH]2)CC1 97996,C#CC1(NC(=O)C(CC(C)CC)NC(c2coc(C)n2)=O)CCCCCC1 97997,N12CC3C(C3C1)C2=O.C(=O)(CCCCN1CCCC1)NC1C(c2ccn(C)n2)C1 97998,c1(CC)c(C(=O)NC2CC(N(C(=O)CC3CC(C)=NO3)C)C2)cccc1C 97999,C1(NC(CSc2ccc(C)cc2C)=O)C2CC3CN(C(=O)C(C)(F)F)C1C3C2 98000,c1(C(=O)NC(c2cn(CCOCCO)nn2)CCC)cc2cccc(Br)c2o1 98001,c1(COC(C)(C)C)cc(C(=O)NC2CCC2NC(c2csnn2)=O)no1 98002,C(=O)(C(C#N)CC1CC1)NCC(C)(C)NC(C1CC(CCC)C1)=O 98003,c1(CC(=O)NC2C(NC(Cc3cc(C)ns3)=O)COC2)cccc(C(C)C)c1 98004,C1(NC(c2c(OC)cc(C)cc2)=O)C(C)CCN(C(=O)C(C)C2CCOC2)C1C 98005,C1(CC)CCNCC1.c1(Cn2ncnc2C(C2CCCCN2)C)nn(C)cc1C 98006,c1(C(=O)NCC2CC(NC(C=C(C)C(C)C)=O)C2(C)C)ccc2c(n1)OCCO2 98007,C1(C(N(CC(CC)NC(c2cscc2C2CC2)=O)CC)=O)CCC(C)(C)C1 98008,Cc1cccc(F)c1CNC(C1CCCN(C(C2CC2C)=O)C1)=O 98009,CCC(C)(CO)C(=O)NCc1cccc(CNC(C2CC3(C2)CC3(F)F)=O)c1 98010,c1(C(N2C(Cn3cc(CNC=O)nn3)CCC2)=O)ccc(S(F)(F)(F)(F)F)cc1 98011,CC1CC2(CCN(CC3CCCS(=O)(=O)C3)CC2)CN1C(=O)CCS(N)(=O)=O 98012,N1(C(C(C)CF)=O)CC2CC(NC(=O)CSCc3ccccc3Cl)C1C2 98013,N1(C(C2CC3(CCCC3)C2)=O)CCCN(C(=O)CN2CCCCC2)C(CO)C1 98014,C1(N(CC(C)(O)C2(C)CC2)C(C2CCCC2)=O)CC(=O)N(O)C1 98015,CC(c1ccccc1)=CC(=O)NCCNC(C1CC(C(F)(F)F)C1)=O 98016,c1(COC)csc(C(=O)NCC2(CO)CN(C(=O)C(F)=C(C)C)C2)c1 98017,C(=O)(CCC(=O)CCC(=O)c1cccs1)OC(c1ccc(OC)c(OC)c1C)=O 98018,C12(CNC(C3CC(C)(O)C3)=O)CCC1CCN2C(=O)CCc1ccccc1Cl 98019,C1(NC(c2cccc(C)c2)C)CCCCC(O)CNCC1 98020,CC1CN(Cc2ccc(-c3ccc(F)cc3)s2)CCN(C)C1 98021,S(=O)(=O)(c1ccc(NCC2(C)CCN(C)C2)c(Cl)c1)N1CCC2(CC(OC)C2)C1 98022,C1(NC(C2C(CCC)C2)=O)CCC(N(C(=O)Cc2cnn(C)c2C)CC)CC1 98023,c1(C(=O)NC(CNC(c2c(C)ocn2)=O)C(C)C)cnc(OCC2CC2)c(Cl)c1 98024,C12(CNC(c3cc4sccc4s3)=O)CCC1CCN2C(c1ccc(F)c(O)c1)=O 98025,CC(=O)CCCC(=O)NC1CC(C)(C(=O)NCCc2noc(=O)n2C)C1 98026,c1(C(N(CCN(C(=O)C(C)(CC)CC)CC)CC)=O)ccc(Cl)nc1OC 98027,N1(C(C2N(C)CCCC2)=O)CCC2(CC(NC(c3cc4n(c3)CCOC4)=O)C2)C1 98028,c1(OC)cc(N(C)CC2CCN(C(=O)CC3COC(=O)C3)C2)nc(OC)n1 98029,c1(C(N(C)CCNC(c2ccc(=N)[nH]n2)=O)=O)ccc2oc(O)nc2n1 98030,C1(C(N2CC(CC)(CC)C2)=O)(CF)CCN(C(=O)CC2CC2COC)C1 98031,C1(CC=C)(NC(=O)CCCNC(C)=O)CC2CCC(C1)N2C(c1cnn(C)n1)=O 98032,CC(C)C(F)(F)CC(=O)N1CCN(C(C2CC(CC(F)(F)F)C2)=O)C(C)C1 98033,N1(C(=O)CCc2nc[nH]n2)CCN2C(=O)NCCC2C1 98034,C(=O)(CCN=C(NCc1cccc(C)c1C)NCC12CCCC(C1)OC2)NC 98035,CC1CN2CCCC2CN1C(C1CC(C)(C)CCN1C(=O)CCC(F)(F)F)=O 98036,C(=O)(CCC(CC)OC)NC(CCCNC(C1(COCC)CCC1)=O)C 98037,c1(CC)ccc(OC)cc1C(=O)NCCCC1CCCCN1C(=O)COCCF 98038,N1(C(C2=C(C)OCC2)=O)CC2CCC(C1)C(NC(C1CC3(C1)CC1(CC1)C3)=O)C2 98039,Cc1ccc(-c2ccsc2C(=O)NC2CN(C(c3cc(C)nn3C)=O)C2)cc1 98040,c1(C(C)C)ncncc1C(N1CCN(CC(C)NC(=O)CC2(C#N)CC2)CC1)=O 98041,C1(CNC(c2cn(C(C)C)nn2)=O)C2CN(C(=O)C(CO)N(C)C)CC12 98042,C1(NC(CC(C)C)=O)CC(NC(c2ccc(O)c(C(C)C)c2)=O)C12CCOCC2 98043,C1(NC(=O)CCN2CCOCC2=O)CN(C(C2CC3(C2)CC32CC2)=O)CC12CC2 98044,c1(C(=O)NC2CN(C(c3c(C)cc(N)cc3)=O)CC2F)cccc2c[nH]nc12 98045,C1(NC(Cc2ccc(OC)cn2)=O)CCN(C(=O)CN2CCCCCC2)CC1C 98046,c1(C(=O)NC(C)COC2CN(C)C2)ccc(N=NC(N)=O)cc1.C1CC1 98047,CC(C)C(C(=O)NCCOC1CC1)C(C)NC(C1CC(F)(CF)C1)=O 98048,C=CCC(C)(CC)C(=O)NCC(C)CN(C)C(c1cccs1)=O 98049,N1(C(CNC(C)=O)=O)CCOC2(CCS(=O)(=NC(=O)C3(C)CC(C)=NO3)CC2)C1 98050,C1(N(C(=O)OCCCC(C)C)C(C)=O)CCC(=O)N(C)C1.CCCCn1cncn1 98051,CCC(C)(O)C(=O)NCC1(O)CCN(C(=O)Cc2ccc(C(F)F)cc2)C1 98052,CC(C)C(F)(CNC(C1(Cl)CC1(F)F)=O)C(=O)N(C)CC1CCCCCC1 98053,N1(C(CC(C(C)C)C)=O)CCC(CNC(=O)CCCCN2CCCC2)C(F)(F)CC1 98054,C1(C(=O)NC2(C(=O)NC3C(C#N)CCC3)CC(CO)C2)Cc2ccccc2C1 98055,CC(=O)CCC(=O)N1CC(NC(c2cc(-c3cccc(Cl)c3)ns2)=O)CC1C 98056,c1(C(=O)NCC(C)CN(C)C(c2csnn2)=O)cncc(-c2cccc(F)c2)c1 98057,C1(C(=O)NCC2N(C(C(C)(C)C(N)=O)=O)CCC2)CN2CCCC2CO1 98058,C1(CNC(Cc2c(C)cc(F)cc2)=O)CCC2CN(C(=O)Cn3cnnn3)CC12 98059,N1(C(C(CC)C2CCOCC2)=O)CCC(N(C(=O)C=Cc2ncc[nH]2)CC)CC1 98060,C(=O)(C1CCCn2nccc21)NC(C1CN(C(c2ccc(=O)n(CCO)c2)=O)C1)C 98061,N1(C(C=C(C)C)=O)CC(CCO)(NC(C2(C3CCCCO3)CC2)=O)C1 98062,C1(NC(N(C)Cc2nnc(O)o2)=O)CNC(=O)C12CC2 98063,N1(C(c2c(C(C)C)con2)=O)CCC(CNC(C2OCCCC2(C)C)=O)CC1C 98064,C(=O)(C#CC1CCCOC1)N1C(C2(NC(C3ON=C(C)C3)=O)CC2)CCCC1 98065,c1(COC)cc(N2CCCC(C3CCCCN3C(C3CC3C(C)O)=O)C2)ncn1 98066,N1(C(c2c(C)[nH]nc2CO)=O)C2CCC1CC(C(N1CCCC(C)(N(C)C)C1)=O)C2 98067,Cc1noc2ncc(C(N3CC(CNC(c4cc(F)cc(Br)c4)=O)C3)=O)cc12 98068,C12(C(=O)NCCC3CN(C(COCC=C)=O)CC3C)CCC(N(C)C)(CC1)CC2 98069,C1(C(N(C(c2cc(C)on2)C)C)=O)CN(C(c2cccnc2O)=O)CC(C)(C)C1 98070,C1(C(=O)NCc2c(OC)nsc2)C(C)OCCN1C(=O)CC1CCN(C)C1=O 98071,N1(C(c2c(C)cc(CO)o2)=O)CC2(CNC(=O)C(C3CCOCC3)O)CCC1C2 98072,c1(C(C)NCC2C(C)CN2C(=O)OC(C)(C)C)nc(N(C)C)co1 98073,N1(C(C2(COC)CCC2)=O)CCC2(CC1)CC2CNC(=O)C(C)CC(C)C 98074,N1(C(C23CCCC2CC3)=O)Cc2cc(Cl)ccc2CC1CO 98075,C1(CNC(C=CCC)=O)(CO)CCCN(C(=O)C(C)OCCCCCC)C1 98076,c1(C(=O)Nc2cccc(CNC(=O)CCc3nncs3)c2)c(F)ccc(F)c1Cl 98077,O=C1OC(CNC(c2cccs2)C2CC2)CCC12CC2 98078,c12cccc(c1)CCC(=O)OC1CN2C1.C1(C(=O)OC)C2COCC12 98079,C1(NC(C(C)C2CCOC2)=O)(CF)CCN(C(C2(F)CC2)=O)C1 98080,C(=O)(CCC(F)(F)Cn1cc(CC(O)C2CC2)nn1)NC(c1cc(Cl)sc1Cl)C 98081,C12(CNC(c3cn(CC=C)nc3)=O)CCCC1CN(C(c1ccc(Cl)cn1)=O)C2 98082,C1(CC(=O)NCCC(=O)NCC#C)CCCN(C(=O)C(C)N(C)CC)CC1 98083,C=CC1(C(N2CCC(O)(CC(C)C)C2)=O)CCN(C(c2ccc(Cl)o2)=O)C1 98084,c1(C(=O)NCCCNC(=O)C=CCN2CCCC2)c(Cl)csc1Cl 98085,CC1(C)CC(CNC(=O)Cn2cccn2)N(C(C2CCC(C)(C)O2)=O)C1 98086,C1(C(N2CCC(NC(C(C)=C3CCC3)=O)C2C)=O)CCOC2(CCC2)C1 98087,C(CCN(C)C)(C(=O)NC1COCCC1O)NC(C1C(C)CC1)=O 98088,CCCC(CCCNC(=O)Cn1nc(C)n(C)c1=O)NC(c1cc(C)[nH]c1C)=O 98089,c1(N)cc(=N)[nH][nH]1.C(C(C)(C)O)N1C(=O)CC2(CC2)C1.CCO 98090,C(=O)(C(C)C(F)(F)C(F)F)NCC(CNC(c1ccc(C(C)C)nc1)=O)(C)O 98091,c1(C(=O)OCc2nc(C(C)OCC)sc2)ccc(O)c2c1CCCC2 98092,c1(NCC(C)N(C)C)ccc(S(=O)(=O)N2CCOC(C3CCOCC3)C2)cc1Br 98093,N1(C(c2cc(CNC(=O)Cc3cnoc3)no2)=O)CC2CCC(CC2)C1 98094,N1(Cc2cn(C(C)C(=O)N3CCC3CC3CCOCC3)nn2)CCCCCC1 98095,C1(NC(C(N2CCC(C)CC2)=O)=O)CC2CCC1N(C(=O)C(C)C(C)O)C2 98096,CCC(C)(C)C(C)CC(=O)N1CC(NC(c2cc(C(F)(F)F)n(C)n2)=O)C(F)C1 98097,C(=O)(CCCN(C)N=O)N1C(C(C)NC(C2CC3C(C2)C3(F)F)=O)CCC1 98098,CC(C)(CN=c1ccnc(C2CC2)[nH]1)NC(=O)CCCCc1cnn[nH]1 98099,c1(N2CC2C)ccc(Cl)c(Cl)c1.c12ccc(cc1)C(n1cccn1)N2C(C1(C)SCCS1)=O 98100,O(S(=O)(=O)c1cc(Br)ccc1Br)c1ccc(-c2ccc(OC)cc2)cc1OCC 98101,N1(C(c2csc(CO)n2)=O)CC2CCCCC2(C2CCCN2C(C2CC2)=O)C1 98102,N1(C(C(C2CC2)OC)=O)CCCC1C1CCN(C(C2CC(C(F)(F)F)C2)=O)C1 98103,Cc1c(Br)noc1C(N1CCC(O)(CN(C(=O)C(O)C2CC2)C)C1)=O 98104,S(=O)(=O)(c1c[nH]ccc1=NCC1CCS(=O)(=O)N1C)N(C)CCn1ccnn1 98105,C1(C(=O)OC(C)(C)C)C2CCC(C2)N1C(c1cnc(C2CCCO2)s1)=O 98106,c1(CC(C)C)cc(C(=O)NC(C2CCOC2)CNC(C2CC(O)C2)=O)no1 98107,C1(C(=O)NC(C)CC2CN(C(=O)C=CC(N)=O)C2)CCC2CCCCN12 98108,C1(C(=O)N(CC(F)(F)F)CCO)CCCN1C(=O)Cc1ccccn1 98109,c1(C(NNC(C2COCCN(C(C)=O)C2)=O)=O)ccc(Cl)c(Cl)c1F 98110,c1(C(=O)NCC(C)CN(C)C(C2CC(F)(CF)C2)=O)c(C#N)ncn1C 98111,C1(NC(c2cc([N+](=O)[O-])c[nH]2)=O)CC2CCC1N(C(=O)Cc1ccno1)C2 98112,c1(C(N(CCC(C)NC(c2ccc(C3CC3)o2)=O)C)=O)ncccc1Br 98113,C(CC1CC1)(CC(=O)NOCC1(C)CC1)NC(C(c1n(C)ccc1)=O)=O 98114,c1(C2N(C(Cn3cc(CCCC)nn3)=O)CCC2)cccc(Br)c1 98115,C1(CC(N2CCC(CCNC(=O)CN3CCCNC3=O)C2)=O)CC2C=CC1CC2 98116,N1(C(CCOCC#C)=O)CCCC(CCNC(c2cc(CC)[nH]n2)=O)C1 98117,Cc1nc(NCc2n[nH]c3c2CCC3)cc(=NCCc2nccn2C2CC2)[nH]1 98118,C=CC1(CC(N2CC(CC)(CC)C2)=O)CN(C(C2CCC2C#N)=O)C1 98119,C1(CN(C(=O)Cn2cccn2)C)CCCN1C(C1(CF)CC1)=O 98120,Cn1ncc2c(NCC3CC3(F)F)nc(N3CC4C5CCC(C5)C4C3)nc12 98121,C#CCCCC(=O)NC1CC=CCC1C(=O)NCc1nnc(O)n1CC 98122,c1(C(=O)NC2C(C(N3C(CC=C)CCCC3)=O)CCCC2)cc2cccnc2[nH]1 98123,c1(C(=O)NCC(CC=C)NC(=O)COC(C)(C)CC)ccc(C(F)F)c(F)c1 98124,Cc1cc(C(=O)NC2CC3(C2)CC(Nc2cc(Cl)nc(C)n2)C3)cc(O)n1 98125,CC1CC=C(C(=O)N2CC(C)(C)CC2CNC(c2sccc2C(C)(C)C)=O)CC1 98126,C1(CNC(c2c(OC)ncc(C)c2)=O)CCC2(CN(Cc3csc(Br)c3)C2)O1 98127,N(C(=NCCC1(O)CCC1)NCC1C2(CC2)C12CC2)C(c1ccccc1)C 98128,C1(CNC(c2c(Cl)nn(C)c2Cl)=O)CC2(CO1)CN(C(C1CCS1(=O)=O)=O)C2 98129,C1(CNC(C2(N=[N+]=[N-])CC2)=O)CCC2(CCN(C(=O)CNC(=O)C3CC3)CC2)C1 98130,Cc1ccc(C(=O)NC2CN(C(c3ccccc3N(C)C)=O)CC2O)n1C 98131,N1(C(c2cn(CC=C)nn2)=O)CC(C(N2CC(F)(C#N)C2)=O)C2(CC2)C1 98132,C1(CNC(c2cnn[nH]2)=O)CCCCCN1C(=O)C=Cc1cc(Cl)sc1Cl 98133,C1(C(N2CC(F)(CNC(CC3C(C)C3(F)F)=O)C2)=O)CC(O)CN1C 98134,c1(NC(c2ncccc2Br)c2n(CCSC)nnn2)ccc(C)c(C)c1 98135,CC1CC2(CO1)CN(C(=O)CCN(CCO)C(c1coc3c1COC3)=O)C2 98136,c1(C(N(C(CNC(c2n(CC)ncn2)=O)C)C)=O)cc2c(cc1N)OCO2 98137,c1(C(N2CCCC(NC(CCCC#C)=O)C(F)C2)=O)c(C)nn2cccnc12 98138,c1(NC(=O)NC2CCc3c[nH]nc3C2)nc2ccccc2cc1[N+](=O)[O-] 98139,C=CCCC(C)(C)C(=O)N1CC2CC2(CNC(c2ccnc3[nH]nnc23)=O)C1 98140,c1(CC(=O)OC(c2ccc(OC)cc2)CC)c(F)cccc1F 98141,c1(C(=O)NCC2C(CNC(c3ccc(SC)cc3)=O)C2)cc(C2CC2)nc(Cl)c1 98142,C1(NC(C(CCCCC)O)=O)CCCCC12CCN(C(=O)CC1(O)CCCC1)C2 98143,C(=O)(CC(C)C(C)(C)C)NC(C1CCCC1)CNC(c1nc(CC)sc1N)=O 98144,c1(OC)cc(C(=O)NCC2(O)CN(C(c3cc(Cl)ccc3I)=O)C2)cc(Cl)n1 98145,C1(C(N(CC(Cl)Cl)C)=O)C(NC(c2ccccc2)=O)C1(C)C 98146,CC1CC(C(=O)NCCN(C2CCCC2)C(c2cncc(F)c2)=O)C(=O)O1 98147,N(C1CC(C)n2ncnc21)C(C1CCCN(CCCOC(C)C)C1)=O 98148,C1(NC(Cc2nc(C(C)C)on2)=O)CC(F)CN(Cc2ncccc2C(F)F)C1 98149,c1(-c2ccc(C(C)O)cc2)cnc2ccc(C(=O)Nc3cncs3)cn12 98150,N1(C(C2C(CCOC)C2)=O)CC(C(=O)NOCC(O)C(C)C)CCC1C 98151,CC(CN(C)C)CC(=O)NC1(CNC(c2cnc(C3CCC3)s2)=O)CCC1 98152,N1(C(CCC#CC)=O)CCC(CCNC(=O)CSS(C)(=O)=O)C(F)(F)CC1 98153,N1(C(c2cnc(CC)s2)=O)C2CCC1CC(CC(C)NC(C1CC13CC3)=O)C2 98154,C(C(C)(C(=O)N(CC(C)CNC(c1cn(-c2cccnc2)nn1)=O)C)OC)OC 98155,c1(CC)ncncc1C(N1CCN(C(CNC(C2CC(O)C2)=O)C(F)F)CC1)=O 98156,c1(SC)ccc(Cl)cc1.C(=O)(CCCOC(=O)C1n2c(cnc2)C(=O)O1)OC 98157,C(CCCC(=O)N(C(C)CNC(c1cccc(OC)c1)=O)C)OC 98158,C(C(=O)Nn1cnn(C)c1=S)N1CC2(N(C(CCCC#CC)=O)CC2)C1 98159,N1(C(c2c(C)c(O)ccc2)=O)Cc2ccccc2C1C(=O)NC1CNC(=O)C1 98160,CC1CN(C(C2(O)CC3CCC2C3)=O)CCC1CNC(=O)CC1CCCCC1O 98161,C1(C(=O)NCCCN(C(C2N(CCC)C(=O)CC2)=O)C)CC2(CCCCC2)CO1 98162,C1(C(=O)NCC(CC)NC(c2c(CNC)noc2)=O)NC(=O)NC1=O 98163,c1(CC)nnc(N2CCC(OCCNC(=O)Cn3cnnn3)C2)o1 98164,N1(C(C(CCC2CCC2)NC(C(C(CC)C)N(C)C)=O)=O)CCOC(C)(C)CC1 98165,C(C)(CO)(C(=O)NC1CCN(CCNC(=O)CC2CCC(=O)NC2)CC1)OC 98166,C1(O)(C(N2CC(NC(c3cnc(SC)s3)=O)C2)=O)CCCCCC1 98167,CC1(C#N)CC2(CC(NC3CCC(O)CC3)C2)C1 98168,C1(CC(=O)NCCCN(C(=O)CCc2cnn(C)c2)CC)CCNC1=O 98169,CCOC(C)(C)c1ccc(NC(=O)NCC(=O)OC(C)C)cc1 98170,N1(C(C2C(C(C)(C)C)C2)=O)CC=CC(NC(C2CCCC(O)C2)=O)C1 98171,C=CCCC(C)(C)C(=O)NC1CCCC1NC(=O)C(CC)NC(N)=O 98172,c1(C(=O)NCCNC(CCc2ccn(C)n2)=O)cc(N2CCCCC2)ncn1 98173,N1(C(C(CNC(C(c2ccccc2)OC)=O)C(C)C)=O)CCC12CCC(O)CC2 98174,C1(N(C(=O)CCC2CC2CC2CC2)C)CCCN(C(C2(C(N)=O)CCC2)=O)CC1 98175,C(=O)(CCC(C)(C)NC(=O)C1CC1)N1CC(c2nc(C)[nH]n2)C1 98176,C(=O)(C1CCc2c[nH]nc21)N1CC(OCC)(CNC(c2cnns2)=O)C1 98177,CC(c1ccccc1F)=CC(=O)OC.C1(=O)CCC(C)SCC(=O)CCN1CC(C)O 98178,N1(C(c2cccc(CC=C)c2)=O)CC2(C(=O)N(CC(C)C(F)(F)F)C)CC1CO2 98179,Cc1cc(C(N2C(C(=O)NCC3(CO)CC4CC4C3)CCC23CC3)=O)nc(C)c1 98180,CC1=C(C(=O)NC2CCC2NC(c2cnoc2C)=O)CCCC1 98181,c1(N(CC(CNC(CNC(C)=O)=O)C)C)c(C#N)cnc2c(C)cc(F)cc12 98182,C1(CCNC(C2(NC(C)=O)CCC2)=O)CCCN(C(c2nocc2C(C)C)=O)C1 98183,C1(C(N(C)CC2C(NC(C(C#C)(C)C)=O)CCC2)=O)CCc2nncn2C1 98184,Cc1csc2cc(C(=O)NC3CC3NC(c3cc(F)cc(F)c3)=O)[nH]c12 98185,Cc1cc(Cl)c(C(=O)NC2CCN(C(=O)CCCC(C)O)C(C)C2)cc1C 98186,c1(C(=O)NCC(=O)NC(CC)CNC(c2csnc2C2CC2)=O)ccc(N)cc1 98187,N(C1CCCc2n[nH]cc21)C(C(c1ccoc1)NC(CC(C(CC)C)O)=O)=O 98188,c1(NC(C2C(N(C)C)COC2)=O)ccc(CNC(=O)CN2CC=CC2)c(F)c1 98189,N1(C(C(C)=C(C)C)=O)CCN(C)CC1CNC(=O)C(O)C(F)(F)F 98190,c1(C2(C(=O)NCC3CCN(S(C)(=O)=O)C3)CCCC2)cc(F)ccc1F 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98244,C1(CC=C)(C(=O)NC2CCC(CNC(C3(O)COC3)=O)C2)CCOCC1 98245,C=CC1CCCN(N2CCCC2c2c(F)ccc(Cl)c2F)C1 98246,N1(C(C2CC(O)(CC#C)C2)=O)CCOCC1CNC(c1c[nH]nc1F)=O 98247,CN1CC=CCC1CC(=O)NC1CCCCC1NC(c1ccsc1C(F)(F)F)=O 98248,c1(C(C(=O)NCC2N(C(=O)CC(F)F)CCC(C)C2)=O)c[nH]c2ccccc12 98249,c1(C(=O)NC2CC(NCc3cc(C)[nH]c3C)C2)c(F)c(F)c(O)c(F)c1F 98250,c1(NC(c2ccc(CCC(=O)NC3CC3(F)F)[nH]2)=O)ncc(F)cc1O 98251,NC1COc2c(CN3CC(CO)OCC34CCC4)cnn2C1 98252,C1(OC)CCn2cc(C(=O)NCC3CC3NC(=O)Cn3ncnn3)nc2C1 98253,C=C(C)C(CC(=O)N1CCCC1CN(C(=O)CC1(O)CCC1)C)OCC 98254,c1(CC)nc[nH]c1C(=O)NCCCCCN(C)C(C1CCC(C)O1)=O 98255,C12(C(=O)NCC3OCCN(C(c4ncn(C(C)(C)C)n4)=O)C3)CC(C1)S(=O)(=O)C2 98256,C1(C(NOCCC(=C)C)=O)CCN(C(=O)Cc2cccnc2)CC1O 98257,C(=O)(CS(=O)(=O)CCC(F)(F)F)NCC(C)(C1CC1)NC(C1ON=C(CC)C1)=O 98258,N1(C(C(C=C)O)=O)CC2CCC(C1)N2C(=O)CSc1nnc(S)s1 98259,C(=O)(CC(C)(C)CNC(=O)C=CC1CCCCC1)NCc1c(COC)noc1 98260,CC(CN(C)C)C(=O)NC(C1CCCN1C(=O)C=CCO)C 98261,N1(C(c2c(C(C)(C)C)ccs2)=O)CC2CCCC2(Nc2nc3cccnc3s2)C1 98262,c1(C(=O)NCCCN(C(C2C(CCC)CCC2)=O)C(C)C)c(C)n[nH]c1C 98263,CC1(C)C(CNC(=O)CCCCCNC(=O)CCCC2CC2)CC1(F)F 98264,C1(NC(c2cncc(C)n2)=O)CCSC12CN(C(c1cc(C(F)F)ccn1)=O)C2 98265,C12(CNC(CCC=C)=O)CC(NC(=O)C(COC)NC(C)=O)(CO1)C2 98266,C1(C(=O)NCCC(CCC)C2CC2)CN(C(=O)C(C)(C)C(C)O)CC1(F)F 98267,C(C(C)(C)CN=c1cccc(S(=O)(=O)NC(C2CCC2)C2CC2)[nH]1)OC 98268,N1(C(CC(CC)C(C)C)=O)CCCC2(CCN(CCO)C2)C1 98269,C(=O)(C(C)(C)C)NCCC(=O)NCCN(C(CSCC=C)=O)C1CC1C 98270,c1(C(=O)NCCCNC(c2nc(CCC)sc2)=O)cncc(C(C)=O)c1 98271,c1(C(N2C(CN(C)C(c3cc(Cl)no3)=O)CCC2)=O)cnc(Cl)cc1N 98272,c1(C(=O)NC(CSCC)C(N2CCC(NC(N)=O)CC2)=O)cnc(F)cc1C 98273,C(C(C)CN=c1[nH]c(=NCCS(=O)(=O)CCO)[nH]c2cccnc12)OCC 98274,Cc1ccc(C(=O)N(CC(C)O)CCNC(C2CCCO2)=O)nc1 98275,S(=O)(=O)(c1ccc(NCc2cn(C3CC3)nn2)c(Cl)c1)NCC(CCCCC)O 98276,CN1CCN(C(C2CCCN2C(=O)CC2CCCCC2)=O)CC1C1CC1 98277,c1(N2CC(C(C)NC(c3ccc(N4CCCC4)cc3)=O)C2)ccnc(C#N)n1 98278,C1(O)(C(N2CCC(N(C(=O)C(C)O)CCOC)CC2)=O)CCC(C)CC1 98279,N1(C(C(=O)N(C)C)=O)CCOC2CCN(C(C3SCCCS3)=O)CC12 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98297,C1(C(N2CC(COC)(NC(C3C=CC3CO)=O)C2)=O)CC2CC1CC2O 98298,c1(CNC(=O)NC(C(=O)OCC)CS(C)(=O)=O)ccc2nc(C)oc2c1 98299,c1(C(=O)NCCN(C(C(C=C)(C)C)=O)CC)cc(=O)n2nccc2[nH]1 98300,C1(C(N(C)CCOCCNC(c2cc(C(F)(F)F)n(C)n2)=O)=O)CCC12CCCO2 98301,N1(C(C=C(CC)C)=O)CC(C)(CNC(C2CCCCS2)=O)CC1(C)C 98302,C1(NC(CC(C)OC)=O)CCCC(NC(=O)Cc2ccc(Br)nc2)C1.C1CC1 98303,C(C(CCO)N=c1[nH]c2c(c(=NCCCn3ccnn3)[nH]1)CCCCC2)OC 98304,c1(C(N(CC(N2CCC(N(CC)CC)C2)=O)C)=O)ccc(Cl)nc1OC 98305,C=Cc1cnn(C)c1C(N1CCCC1CN(C)C(C1CC(=C2CCC2)C1)=O)=O 98306,C1(CNC(C2(C#C)CC2)=O)CN(C(c2cc[nH]c2CC)=O)CC12CCC2 98307,c1(CC(=O)NCCC(C)NC(=O)C(c2ccccc2)O)cccc2c1OCO2 98308,Cn1cc(Br)cc1CNc1ccc(C(F)C(F)(F)F)cc1 98309,c1(C(N2C(CNC(c3n(C)ccn3)=O)COCC2)=O)cc2c(Cl)c(F)ccc2[nH]1 98310,c1(C(=O)NCC2CC2NC(C2CC(C(F)(F)F)C2)=O)ccc(F)c2c1OCC2 98311,C1(C(=O)NC(CC)CN(C)C(c2cc(C3CC3)[nH]n2)=O)OCC2CCCC12 98312,C(=O)(CS(=O)(=O)C1CCCC1)NC1C(NC(C(C(CC)CC)OC)=O)C1 98313,C1(NC(CC(C)(C)SC)=O)CC(O)CN(C(c2cccc(O)c2Cl)=O)C1 98314,C1(NC(c2c(C)nc(O)[nH]2)=O)CC2CCC1CN(C(c1csc(=N)[nH]1)=O)C2 98315,c1(C(=O)NC2CCOC2C(N2CC(CO)C2)=O)cncc(O)c1 98316,Cc1nc2cc(CNC(C3CN(c4ncc(C)c(C)n4)CCC3O)=O)cnc2[nH]1 98317,c1(C(C(=O)O)NC(CN(C)C(c2ccc(Br)s2)=O)=O)c[nH]c2cc(F)c(F)cc12 98318,C=C=CC(C)C(=O)NC1(C(N2C(C(=O)OC)CC2C)=O)CC1(C)C 98319,c1(C(N(CCC(C)NC(=O)C(c2ccc(F)cc2F)C)C)=O)cnc(Cl)cc1N 98320,c1(C(=O)NCCC2(CNC(CC(C)c3ccco3)=O)CC2)nccc2ccsc12 98321,Cc1cc(=O)c(NC(=O)C(C(C)NC(c2csc(Cl)c2)=O)C(C)C)c(C)[nH]1 98322,C1(CC=C)(C(=O)NCc2nc(C(N3CCCC3C(=O)NCC)=O)co2)CCOC1 98323,c1(CC)noc2ncc(C(=O)NCC(F)CNC(c3cscn3)=O)cc12 98324,c1(N(C2CC23CCNCC3)C(COC(C)C)=O)ccc(O)cc1O 98325,c1(NC(C(Cc2cc[nH]n2)NC(C(C)=C2CC2)=O)=O)ccc2c[nH]nc2c1 98326,c1(C(N(C2CN(C(c3ccc(C)nc3)=O)CC2F)C)=O)ccnc2ccsc12 98327,c1(C(=O)NC2CC(NC(=O)CC3CCOC3)CC2O)cc2sc(Cl)cc2[nH]1 98328,Cc1cc(O)ccc1C(N1CCC(NC(=O)C(=O)Nc2c(F)cccc2F)C1)=O 98329,C(=O)(CCCCCCNC(=O)Cn1ccccc1=O)NC(C)C(C)(C)O 98330,N1(C(c2ncsc2C(F)(F)F)=O)CC(NC(C2(CO)CC2)=O)C(C(F)F)C1 98331,N1(C(CCN(C(C(C)OCC=C)=O)CC2CC2)=O)CCC(O)(CN(C)C)C1 98332,C1(OC)CC(C(N2CCCCC2CNC(=O)CC2CCCSC2)=O)CC1OC 98333,c1(C2C(=O)N3CCC(C3)CO2)ccccc1.c1(O)ccccc1.CC(C)O 98334,c1(C(C)C)ccc(Cl)cc1C(=O)N(C(C)CNC(=O)Cc1cnoc1)C 98335,N1(CC(CO)OC)CCCC1CNC(=O)CCc1nccn1C(F)F 98336,C(=O)(C1=NOC(CNC(=O)C(O)CN(C)C)C1)NCC1ON=C(C)C1 98337,N1(C(C2N(C=O)CCC2)=O)CCN(C(=O)Cc2c[nH]nc2O)CC(O)C1 98338,C1(C(=O)NCC(c2ccccc2)CNC(CCSC)=O)CC(=O)C12CCCC2 98339,c1(N(C(C(CNC(c2c(C)csc2C)=O)O)=O)C)cccc(F)c1C 98340,O(NC(=O)CC(CNC(=O)CC1CC1)OC)CC#C 98341,c1(CC(=O)NCC(C)NC(c2noc(-c3ccccc3F)n2)=O)cncc(F)c1 98342,O=C(CS(=O)(=O)N1CCOCC1)NCC1CC(O)CN1C(=O)C=CC1CCCO1 98343,C(=O)(CCC(C)(C)F)N1CC(C2N(C(c3cc(C)n(C)c3)=O)CCC2)(O)C1 98344,N1(C(c2n(CC)ncn2)=O)CC(NC(c2ccccn2)=O)C(C(F)(F)F)C1 98345,Cc1cc(=NCC23CC2CN(C(=O)Cc2ccccc2I)C3)[nH]cn1 98346,C=CCC(CNC(=O)CNC(N)=O)NC(C1CCN1C)=O 98347,N1(CCOC)CC(C(=O)NCC2CCC2NC(c2cc(C)ns2)=O)CC1=O 98348,c1(C(=O)NCCN(C(Cc2cc(C)[nH]n2)=O)CC2CC2)cc(C)c(N)cc1F 98349,N1(C(CN(C)C(C2CCC3(CC3)C2)=O)=O)CCC2(C=CCO2)C1 98350,CC1(C)CC(n2nc(Cc3cccc(Cn4cncn4)c3)nc2-c2cnc(Cl)[nH]2)CO1 98351,n1(CC(=O)NC23C(C)OC(CNC(=O)CC#N)(C2)C3)nc2ccccn2c1=O 98352,C(=O)(C(C(C)CC)N(C)Cc1ccccc1Br)NCC(=C)C 98353,N1(C(C2CC3OC2C2CC32)=O)CCC2CN(C(c3ccnc(C(F)F)c3)=O)C2C1 98354,C(CC(C)(C)C(=O)NC1CCC1NC(=O)Cc1ccc(C)cc1)OC 98355,C1(C#N)(C(=O)NC2CCN(C(c3c(Cl)nc(OC)s3)=O)C2)CC12CCC2 98356,N1(C(c2c(OC)nccc2)=O)CCN(C(=O)CN(C2CCSC2)C)CC2(CC2)C1 98357,C1(NC(CC2N(CC)CCOC2)=O)CCN(C(=O)C(C2CCC2)OC)C(C)C1 98358,C1(C(C)C)C2CCN(C(=O)C(C3CCN(C(c4nc(=N)cc[nH]4)=O)CC3)C)CC12 98359,c1(C(=O)NCC(CNC(=O)CC2(CO)CC2)OC)ccc2[nH]c(=N)[nH]c2c1 98360,c1(C(N2C3(CN(C(C4CN(C)C4)=O)C3)CCC2)=O)c(O)cccc1[N+](=O)[O-] 98361,c1(NC(C(CC)O)=O)ccc(C(C)NC(=O)COc2ccsn2)cc1 98362,C1(CNC(c2c(C(C)C)nns2)=O)C2CN(C(C3CCCN3S(C)(=O)=O)=O)CC12 98363,C(=O)(C(CC)C(C)O)NC1(CC=C)CCN(C(=O)CCc2ccc(O)nn2)C1 98364,CCCC(C(=O)N1CC(C)(CCC(=O)NC(c2nccnc2C)C)C1)NC(C)=O 98365,C1(NC(C(CC)C)=O)CCCCCC1C(=O)NCc1ccc(Cl)cc1 98366,N1(C(C2C(=C)C2)=O)CCC2CN(C(=O)CCCOc3ccccc3Cl)CC2C1 98367,C1(C(N2CC3CC3(C(=O)NC3CCC3)C2)=O)CCC(C(F)(F)F)CC1 98368,C(=O)(C1CCCc2nc[nH]c21)N1CCC(C)(NC(c2cccc(N)c2N)=O)C1 98369,C1(C)(C(=O)NCC2=CCN(C(C3CCCC(C)(C)O3)=O)CC2)CCCCNC1=O 98370,N1(C(Cc2c(C)ocn2)=O)CC(NC(C2CC3CC3C2)=O)CC(C)C1 98371,C(=O)(C#CC(C)(C)CNC(C1COCCN1C)=O)NCC1(C)ON=C(C)C1 98372,c1(-n2c(-c3ccc(-c4[nH]cc(C#N)c4)cc3)ncc2)ccc(F)cc1F 98373,C1(CNC(C=CC=CC)=O)CCN(C(c2ncc(C)cc2F)=O)C1(C)C 98374,N1(C(COCCCC)=O)CCN(C(=O)CC2COC(C)(C)CO2)C(C2CCC2)C1 98375,C1(C2CCC2)(C(=O)NCC2C3N(C(C(C(C)C)CO)=O)C(CC3)C2)CC1(F)F 98376,c1(CC(N2CC(C)N(C(=O)Cn3cccn3)CC2C)=O)cc2cc(Cl)ccc2[nH]1 98377,c1(NC2(C)CC(NC(C3(C)CNC(=O)C3)=O)C2)ncc(C(N)=O)cc1Cl 98378,c1(C(N(CC(C)NC(C2C(C#C)C2)=O)C)=O)ocnc1C1CC1 98379,c1(CN2CCC(CC(=O)N(CC=C)CC3CCOC3)C2)c(F)cccc1F 98380,C1(C(=O)Nc2c(CC)n(CC(C)C)nc2)CCC2(CC1)CCC2N 98381,c1(C(N2C(CNC(c3cncc(C)c3)=O)CC(C)(C)C2)=O)cncc2nc[nH]c12 98382,CCC1=C(C(=O)NC2C=CC(C(=O)NCCC(C)(O)C3CC3)C2)CCCO1 98383,c1(C(N(CCCNC(=O)CCCc2cnn[nH]2)C)=O)ccc2oc(O)nc2n1 98384,N1(C(c2ccc(CC)o2)=O)CCCN(C(c2cscc2CC)=O)CC1CO 98385,C1(CCC2CC2)CN(C(c2cn(CCC(C)C)nn2)=O)CCN1C(=O)C(=O)OC 98386,c1(NC(CC2(NCC3N(C)CCCC3)CCC2)=O)c(C#N)ccc2ccccc12 98387,Cc1nc(C(=O)N(CC2CCN2CC)Cc2ccc(N3CCCCCC3)cc2)cn1C 98388,CC1(NC(C2(C)COC2)=O)CN(C(c2cn(Cc3ccccc3)nn2)=O)C1 98389,C(=O)(C1CCCc2ncccc21)NCC1CC(NC(C2CC(C)OC2)=O)C1 98390,C1(CNC(COC2(C)CN(C(c3c[nH]c(C#N)c3)=O)C2)=O)CCCC(F)C1 98391,CCCN=C(NCCN1CCCCC1)NC1CCCC1CNS(C)(=O)=O 98392,c1(OC)cc(CCC(=O)NC2CCCN(C(C3CCOC3C)=O)C2)ccc1Cl 98393,Cc1cc(CNC(c2c[nH]nc2C2CC2)c2nnnn2Cc2ccco2)sc1C 98394,c1(C(=O)NCC(C(C)C)NC(C(CC)N(C)C)=O)cc2ccccc2n1C 98395,CCC(CC)C(=O)NCC1CN(C(=O)C(n2ccc(C)n2)C)CC1O 98396,C=CC(C)CC(=O)NCC(CC1CCCC1)C(=O)NCCOCC(=O)OC 98397,c1(C(=O)Nc2ccc(COC(C3(OC)CCC3)=O)cc2)cccc(C)c1C#N 98398,C1(NC(C2(C#N)CCC2)=O)CCN(C(c2cnc(O)s2)=O)CC1c1ccccc1 98399,c1(N2CCC(C)C2CNC(c2cccc(F)c2F)=O)nc(Cl)nc2nc(Cl)n(C)c12 98400,N1(Cc2c(Br)ccc(C)c2)CC2CC(NC(=O)Cc3c(C)noc3C)CC2C1 98401,C1(CNC(CC2CC(SC)C2)=O)C(C2CC2)CCN1C(=O)Cc1cscn1 98402,C1(C(=O)NCC(CC)N(C(=O)CCC2CCC(C)O2)C)CC(F)(CF)C1 98403,C1(NC(c2c(C(C)(C)OC)cccc2)=O)CC(O)CN(C(=O)C(C)=C2CCC2)C1 98404,Cc1c(Br)ccc(F)c1C(=O)NC12CCC1CN(C(=O)C#CC1CC1)C2 98405,Cc1[nH]c(C#N)cc1C(=O)NCc1cccc(C(N2CC(C)(C)C2)=O)n1 98406,CCC(CC)CC(=O)N1CC(NC(=O)CCc2nncn2C)C(CC(C)(C)C)C1 98407,C1(CNC(C(N2CC3(CN(C(C)=O)C3)C2)=O)=O)CC2CC1CC21CC1 98408,C12(NC(=O)COC3CCC3)CCCN(C(=O)CCCC(F)(F)F)CC1C2 98409,Cc1cc(=NC2CC3CN(C(=O)CC4(C)CCCC4)CC23)[nH]c(Cl)n1 98410,C(c1cnc(O)nc1O)=CC(=O)NC(C)(CNC(c1ccccc1Cl)=O)C1CC1 98411,c1(N2Cc3c(C)cccc3CC2)nc(=NCC(C)CCO)[nH]c2ccccc12 98412,C1(C(=O)NCC=CCNC(=O)C(C)=CC2CC2)(COC)CCCC1 98413,c1(CCCC(=O)NCC(CNC(CNC(CNC(C)=O)=O)=O)O)ccc(O)cc1 98414,C1(C(=O)NCc2ccc(CCNC(c3cnsn3)=O)cc2)(COC)CC=CCC1 98415,C(=O)(C(C)(C)CS(N)(=O)=O)N(CCN(C)C(c1ccc(F)cc1C(F)(F)F)=O)C 98416,Cc1cc(C)c(C(=O)NCCCCC(C)NC(=O)C(C)(C)C2CCCCO2)cn1 98417,N1(C(C(CC=C)CN)=O)CCc2sccc2C1CC 98418,c1(OCC(N2CC(C3N(C(C(C)(C)C)=O)CCC3)(O)C2)=O)cncc(F)c1 98419,C1(C(=O)NCCC)CCN1C(=O)CSc1nc[nH]n1 98420,C1(C)(NC(C2N(C(CS(CC)(=O)=O)=O)CCOCC2)=O)CCCCC1(C)C 98421,c1(OC)cc(C(N2CCCCC2CNC(C2CCS(=O)(=O)N2C)=O)=O)cc(C)n1 98422,n1(CC)cc(Cl)c(C(N2CCC(N(C(=O)CC3CCS(=O)(=O)C3)CCO)C2)=O)n1 98423,C1(C)(CC)CC(NC(c2ccc(OC)c(Cl)c2)=O)CN1C(=O)CCOCC1CC1 98424,N=c1[nH]c2c(s1)CN(c1ccc3occc3n1)CC2 98425,CCCC(C(=O)N1CC2CC1C2NC(C1CCC1c1nc(S)n[nH]1)=O)S(N)(=O)=O 98426,C1(CCNC(C(C)NC(=O)Cn2cnnn2)=O)CCCCN1C(=O)CNC=O 98427,C(C(C)CN=c1nc(N2CCCC3(CCSCC3)C2)c2sccc2[nH]1)OC 98428,CCCCC(C(=O)NCC(C)(C)NC(c1cnnc(O)c1)=O)C(C)C 98429,C(=O)(C1=NOC(C)(C)C1)NC(C(C)C)CC(=O)NC(c1cn(C)nn1)C 98430,c1(SC)cc(C(=O)NC2CC(CNC(C3CC=CCO3)=O)C2)nn1C 98431,c1(C(=O)NCC2CC(NC(c3cc[nH]n3)=O)C23CCC3)c[nH]c2cnccc12 98432,N1(C(C(C(=O)OCC)F)=O)CC2CCC1C1CN(C(=O)C(C)(F)C(C)(C)F)CC21 98433,C(C(C(C)C(C)C)Nc1ncns1)NC(CCc1cncc(OC)c1)=O 98434,C1(c2c(C)cccn2)CCN(N2CCN(C(=O)C(C)(C)C)CC2)C1 98435,n1(CC2CC(NC(C(C(C)C)N(CCOC)C)=O)CN2C)cnc2ccccc12 98436,c1(N2CC(C)(CCO)OCC2)ccncc1S(=O)(=O)NCC(C)(C)c1cccs1 98437,c1(C(NOCC(=O)NC(CC#C)C)=O)ccc(O)nn1 98438,N12CC3COCC(C1)(C3O)NC(=O)C2.N1(CCO)CCN(c2cccnn2)CC1 98439,CC(O)(Cn1ccccc1=O)C(=O)NC1CC(F)(CNC(=O)Cn2cncn2)C1 98440,Cc1ccc2c(=NCC3CCOCC3)[nH]c(=NCCC(C)(C)CO)[nH]c2c1.C(C)C 98441,N1(C(CCC=CC(C)C)=O)CC(NC(c2ccccc2Br)=O)CC2(CC2)C1 98442,N1(C(C2(C(C)NC(=O)CC3C=CCCC3)CC2)=O)CCC(C)(CO)CC1 98443,O=C1CNc2cc(C(N3CC4CC3CN(C(=O)C3=CCOCC3)C4)=O)cnc2N1 98444,N1(C(C(COC)NC(C)=O)=O)CCN(C(=O)C(O)CC(N)=O)C(C)C1 98445,N1(C(CC(COC)C)=O)CC2CCCC(C1)N2C(=O)C(CC(F)F)C1CCC1 98446,N1(C(C2C(C)CC(=O)C2)=O)CCN(C(c2cnn3ncccc23)=O)C2(CCC2)C1 98447,C1(CC(=O)NC2C(CNC(C)=O)C2)(NC(=O)CSC2CCCCO2)CCCCC1 98448,CC(C)C(C)C(=O)NC1(CCNC(=O)C(c2ccc(F)cc2)O)CCCC1 98449,C(C(=O)NCCN(C(=O)C(c1cscn1)N(C)C)C)(OCC)OCC 98450,c1(C(=O)NC2CN(C(=O)C(F)CC3CCCCC3)CC2CO)ncc(Cl)cc1O 98451,N1(C(C(CC#C)(C)NC(=O)C(c2ccn(C)n2)C)=O)CCN2CCCC2C1 98452,Cc1cc(C(N2CCCC(C3CCCCN3CCn3nccc3N)C2)=O)sc1C 98453,C1(NC(c2cc(OCC(F)(F)F)ccn2)=O)CCCC(NC(C2C=CCC2)=O)C1 98454,C1(C(N)=O)CCCN(CCC(=O)NC2CN(C(C3CCN(C)CC3)=O)CC2O)C1 98455,n1(CC)ncc(C(=O)NC2CC(NC(=O)CCC3CCCCN3C)C(O)C2)c1C 98456,C1(CN(C(=O)C(C)N(C)CCN(C)C)CC(=C)C)C2CCCC12 98457,N1(C(c2cn(CCOC)nc2)=O)CCC(CCN(C(=O)C(C)SC(C)C)C)CC1 98458,C(CCN=c1nc(N2CCC(C)C3(CCCCC3)C2)cc(C)[nH]1)OCC 98459,C#Cc1ccc(F)c(C(=O)N(C2CCN(C(=O)C=CC(C)C)CC2)CCO)c1 98460,c1(C(N2CC(CCCNC(C(CC)OC)=O)OCC2)=O)cc(F)ccc1C1CC1 98461,CCC(CNC(c1ccc2cc[nH]c2n1)=O)(CC)C(=O)NCC1CCOC1C(C)C 98462,CC1CN(C(C2COC(=O)N2C)=O)CCN1C(C1CN(S(=O)(=O)C(F)F)C1)=O 98463,C1(NC(c2c(OC)csc2)=O)CCN(Cc2c(C)noc2C)CC1(C)C 98464,CCC(CC(=O)N(CC(O)CNC(c1ccn(CC)c(=O)c1)=O)C)C(F)F 98465,c1(C(C(=O)NCC2N(C(C=CC=CC)=O)CC=C2)C)ccc(SCC)cc1 98466,c1(C(c2nnnn2CC2CC2)NC(C)C(=O)NCCF)cc2nc(Cl)ccc2s1 98467,c1(CNC(=NC)NCCC(C)CCC(=O)NC)nnn(C)c1N 98468,C1(C(N2CC(CCCCNC(C(C)=C(C)C)=O)C2)=O)C2Cc3cc(Cl)ccc3C12 98469,N1(C(C(C)SCC)=O)CCOC(CCNC(C2(c3cccnc3)CCCC2)=O)C1 98470,C1(NC(C(=O)NCCc2ccc(OCC)cc2)=O)CCCCC1(OC)OC 98471,N1(C(Cn2c(C)nc(C)n2)=O)CCC(C(=O)NCCc2nncn2C)CC1(C)C 98472,N1(C(C2ON=C(C)C2)=O)CC2CN(C(c3cc4cnccc4o3)=O)CC2(C)C1 98473,C1(NC(CC=C)=O)CCN(C(c2occc2C)=O)C1C(C)(C)C 98474,C1(C(=O)NC2C(CNC(c3nc(C)c(C)s3)=O)COC2)CCC(=O)N(C(C)C)C1 98475,c1(N(C(C)=O)C)cccc(C(=O)NC2CCC(NC(c3cncs3)=O)CC2)c1 98476,CC(CC(=O)N1OCC(F)(F)C(=O)NCC(C)C1)C(C)(C)C 98477,CC(CC(=O)N1CC(NC(c2cccc(Cl)c2)=O)C1)C(=O)c1ccccc1 98478,c1(NC(C(CCC)N(C)Cc2cn3ccsc3n2)=O)cnc(C)c(C#N)c1 98479,CCCCCCCCCCCC(=O)NCC1CCCN(C(C2CCSC2)=O)C1 98480,c1(C(=O)NC2CC(CCC(=O)NCCC(C)(C)OC)C2)c(C)nsc1N 98481,c1(C(N(CCNC(C(CC)SC)=O)CCOC)=O)nc(C)ncc1Br 98482,C1(NC(c2cnc[nH]2)=O)CN(C(=O)CC2CC3(CC3)C2)C2(CCOC2)C1 98483,C1(NC(C(C)OCCC=C)=O)CCCC12CCN(C(c1cc(Cl)sc1Cl)=O)CC2 98484,c1(C(N(C2CCCN(c3ncnc(Cl)c3CO)C2)C)=O)ccn2nccc2n1 98485,N1(C(C(c2cn(C)nn2)NC(C2C(CC)C2)=O)=O)CC(F)(C2CC2)C1 98486,N1(C(C(=O)NCC)=O)CCOCC1CN(C(=O)C(C)(C)c1cncs1)C 98487,C1(c2nc(C(C3CC3)OCC)nn2-c2ccc(C)c(C)c2)CC2(CCOC2)C1 98488,N1(C(C(c2scc(C)n2)C)=O)CCC2(CCC(CNC(C34CC3C4)=O)OC2)CC1 98489,c1(C(=O)NC(C)CNC(=O)C=Cc2c[nH]cn2)cnc(C(F)(F)F)nc1 98490,C(=O)(N=c1nc(C2CCCCCC2)[nH]s1)Nc1cc(C)n(-c2ccccc2)c1C 98491,Cc1cc(N2CCCC(C)C2CNC(=O)C(C)(C)CC(C)(C)C)ncc1[N+](=O)[O-] 98492,c1(OC)c(NC(C2CCN(Cc3c(F)ccc(C)c3Br)CC2)=O)ccc(F)c1F 98493,N1(C(C(C)OCC(C)C)=O)CC2(C=C(C(=O)NCc3nn[nH]c3C3CC3)CO2)C1 98494,N1C(CC(=O)Nc2nn[nH]n2)CCOCC1=O.C12(CCC1)CC(=O)OC2C(C)(C)C 98495,C1(NC(CC(C)C)=O)C2CN(C(=O)C(N3CCC(O)CC3)C)CC12 98496,c1(N(C2CNC2)C(c2n(C)nnc2)=O)ccn2ncc(Br)c2n1 98497,C1(CNC(c2ccc(OC)s2)=O)CC(C)(C)CCC1NC(=O)C(C)(C)CC(C)C 98498,C(=O)(C1=CCCCC1P(C)(C)=O)NC1C(CNC(C(C)(C)c2ccccc2)=O)C1 98499,c1(C(=O)NC2C(CNC(c3ccnc(C(F)F)c3)=O)C2)cncc2cnccc12 98500,N1(C(c2c(C)cco2)=O)CCC(C(=O)NOCCN(C)C)C12CC2 98501,C1(NC(=O)COCC2CCCO2)CCCC(NC(=O)Cc2nccc(O)n2)C1 98502,N12CCC3CCCC13C(=O)OCC(O)CC2=O.N1(C(=O)OC(C)(C)C)CCCC1 98503,N1(C(CCCCOC)=O)C2CCC1CC(NC(=O)C(C(C)(C)C)NC(C)=O)C2 98504,CCC(CC)CC(=O)N1CC=CC(C(=O)NCC=CC(=O)OCC)C1 98505,N1(C(c2n(C)nc(C(F)F)c2)=O)CCC(NC(C2CC2(C)C)=O)C12CCC2 98506,N1(C(CCCC(=C)C)=O)CCCC(C2CCN(C(C3CN4CCN3CC4)=O)C2)C1 98507,c1(C(N2CCN(Cc3nc(Cl)ccc3F)C3CC23)=O)cnn2cccc(F)c12 98508,c1(N(C(=O)OCC)C)ccc(NC(C2(c3ccccc3Cl)CCOCC2)=O)cc1 98509,c1(C(=O)NC(CC(C)NC(C=CCC)=O)C)c(C)sc(C)c1Br 98510,CC1CCCN(C(c2cnc(Cl)s2)=O)C1CNC(C1C2COCC12)=O 98511,C(C(C)CC(F)(F)F)NC(C(c1ccnn1C)NC(C(C)SCCOC)=O)=O 98512,C1(C(N(c2sc3cc(C)sc3n2)C)=O)Cc2ccccc2CN1CC#N 98513,Cc1cc(Br)cc(C(N2CCC(O)(C(=O)N(C)C)CC2)C(=O)NC2CCCCC2)n1 98514,c1(C(=O)OC)ccc([N+](=O)[O-])c(N2CC3CC(NC(c4ccc(C)[nH]4)=O)C3C2)n1 98515,c1(NCC)cccnc1C(=O)NCC1CCC1NC(C1(n2cccn2)CC1)=O 98516,O(N=C1CCCCCC1)CC(=O)NC1CN(C(C(CCC)C)=O)CC1C(F)(F)F 98517,C1(NC(c2ncn(C(C)C)c2)=O)CCOCC1NC(=O)CC(=O)NC1CC1 98518,C1(C(C)NC(=O)C(C)n2cccn2)CCN(C(c2ccnnc2Cl)=O)CC1 98519,c1(CC)ccc(F)cc1C(N1CCC(NC(=O)C(F)(F)c2cncs2)C(O)C1)=O 98520,C#Cc1cccc(CC(=O)NCC2(NC(c3ncccn3)=O)CCCCC2C)c1 98521,C1(C(=O)NCC=CCC(=O)N(CC(N)=O)CC)CCSCC1 98522,O=c1cc(NC2COC(C(F)(F)F)C2)[nH]cc1I 98523,c1(OC)ccc2c(c1)OCC(C(=O)N1CCN(C)C3(CC3)C1)=C2 98524,N1(C(c2cnc(C(C)C)s2)C(=O)NC)CCN(C(=O)OC(C)(C)C)CC1C 98525,c1(C(N(C2CCN(C(c3cc(C)on3)=O)C2)CCO)=O)cc(N)cnc1C 98526,O=C1NC(=O)C2(CCN(C(=O)NC(c3ccc4ccccc4c3)C(F)(F)F)C2)N1 98527,O=C(C1=CCCC1)NC1CN(c2cc(-n3cncn3)ncn2)CC1F 98528,C(c1c(F)cccc1F)=CC(N1CC(OCCNC(C(C(C)OC)O)=O)C1)=O 98529,c1(CNC(C(CC)=CCCC)=O)ccc(CNC(=O)CCc2cnccn2)cc1 98530,Cc1cc(C(N2CCCC(C(C)NC(=O)CCF)C2)=O)cc(I)c1 98531,c1(OC)ccc2c(c1)CCN(c1ccc(S(=O)(=O)NC3CSC3)cc1F)C2 98532,N1(C(C(CC)Oc2ccccc2)=O)CCC2CN(C(c3ccn(C)c3)=O)C2C1 98533,C1(C(N(CCCCCNC(C(COC)N(C)C)=O)C)=O)OCCOC1(C)C 98534,c1(C(=O)NC2CC3(C(NC(c4c(N)cc(Cl)nc4)=O)C3)C2)n[nH]c2c1CCSC2 98535,C1(C(=O)Nc2cccc(CNC(CCCC#C)=O)c2)CCn2c(C)cnc2C1 98536,c1(C(=O)NCC(CC=C)NC(C2CCC(CO)CC2)=O)cc(C#N)ccc1F 98537,C(CCCCCC(=O)N1CCC(O)C(F)(F)C1)NC(C1CC2CCC1CC2)=O 98538,CCCCC(C)CCC(=O)NCC1(NC(c2ccc(O)cn2)=O)CCOCC1 98539,n1(CC)c(OCCOC)nnc1N1CCC(CCN2CCN(CC)CC2)CC1.COC 98540,C(N=C(NC1CC1)NC1CC(C)(C)CCc2ccccc21)c1c(C)ncs1 98541,C1(CNC(COCCOC)=O)CCCC2CN(C(c3cccc4c[nH]nc34)=O)CC12 98542,n1(CC(N2CCC(CN(C(c3c(OC)scc3)=O)C)C2)=O)nc(C)c(Cl)c1C 98543,C(=O)(CCC(C)(C)F)N(CCCCN(C)C(C1CCOC1c1cnn(C)c1)=O)C 98544,CC1(C)CN(C(=O)COc2ccccc2F)CC1NC(=O)CCCCO 98545,CC(C)(C)CC(C)(C)C(=O)NCCN(C1CCCCCC1)C(=O)Cn1[nH]cnc1=N 98546,Cc1ccc(NC(C)CNC(c2sccc2C(C)C)=O)c([N+](=O)[O-])c1 98547,Cc1cccc(C(C)C(=O)N(CCNC(=O)C#CC2CC2)CC2CCCCC2)c1 98548,CCC(C)CCC(=O)NC1CCCCC1NC(=O)Cn1cc(C(=O)OC)nn1 98549,C1(C(=O)NC(CCSC)Cc2ccccc2)CCCCC(C)(C)C1 98550,c1(C(=O)NCCN(CCC)C(c2ncc(F)cc2N)=O)c(Cl)nc2ccccn12 98551,c1(C(=O)N(C2CC2)CC2CCCN2C(c2csnn2)=O)coc2c1CS(=O)(=O)C2 98552,C1(C(N2C3C(NC(C(C)OCCOC)=O)C(C3)C2)=O)CCCC2(CCOC2)O1 98553,N(C(=NCCN1CCOCC1(C)C)NCCOC)C(c1cccc(C)c1)C#C 98554,C(=O)(C#CC1CCCC1)NCC(CC=C)C(=O)N1CCSCC1 98555,N1(C(c2cc(SC)oc2C)=O)CCC2(CCC2NC(c2occc2C)=O)CC1 98556,C=CCC(C)C(=O)NC1(C(=O)NCCCn2ccnc2)CC1 98557,Cc1nn(C(C)C)c(C)c1C(=O)NCCCNC(=O)Cc1ccccc1Cl 98558,C1(COC)(NC(=O)Cc2nnc(C)s2)CCCN(C(c2ccc(OC)cn2)=O)C1 98559,c1(C(N2C(CNC(C(CCC)C)=O)CCCC2)=O)c(C)cccc1C 98560,C(=O)(C(O)CC(C)C)NCCCN(C(c1csc(-c2nc(C)cc(C)n2)n1)=O)CC 98561,C12(NC(c3nc(CCOCC)oc3)=O)CCN(C(=O)CNC=O)CCC1C2 98562,c1(N2CCC(O)(c3onc(C(C)C)n3)C2)nccc(Br)c1F 98563,C1(NC(C2CC(C)(CC)C2)=O)CN(C(C2C3CCC(=O)C23)=O)CCC12CCC2 98564,C=CCCC(C(=O)N(C(C)CC(N)=O)C)NC(C1C(C)C1C)=O 98565,N1(C(CCC2C(C)(C)C2)=O)CC2CC(C1)N(C(c1occc1Br)=O)C2 98566,C(C)(C)(C(C)CC(=O)NCC1CC12CC2)NC(CNC(=O)NC)=O 98567,N1(C(C(CCC#C)O)=O)CCN(C(c2ccc(C(F)(F)F)nc2)=O)CC2(CC2)C1 98568,C(C1=CCN(C(=O)CC(F)(F)F)CC1)NC(Cn1c(C(C)C)nnn1)=O 98569,C(=O)(CCCC(F)(F)C(F)(F)F)NC1CCCC(NC(c2nc(C#C)sc2)=O)C1 98570,C1(CN(CC)CC2CCCCO2)CCCOC1c1ncc[nH]1 98571,N1(CCC)CCCCC1CN=C(NC(CC)CC)NC1CCS(=O)(=O)C1 98572,C1(NC(c2cnc(C(C)C)s2)=O)CC2CCC1N2C(=O)CC1CC(=O)NC(=O)C1 98573,c1(C(=O)NC2CCCN(C(c3cccc(SC)c3)=O)C2C)cc2cccnn2c1 98574,C1(SC)CN(C(C2(O)CC(F)(F)C2)=O)CC1NC(C1(C)CC1(F)F)=O 98575,C1(NCc2cccc(-c3nnc(C)o3)c2)CCC(C)(C)CC1C(=O)O 98576,Cc1oc(C)c(CN2CCC(NCCN3CCCCC3)CC2)c1C 98577,C(c1cccc2cccnc12)=CC(=O)NC1(C2CN(C(C(C)(C)OC)=O)C2)CC1 98578,Cc1cccc(C)c1OCCNC(=O)C(N1CCC(C)(CC2CCCCO2)C1)=O 98579,c1(C(N(c2cc(C(C)(C)C)ccn2)CC)=O)cc(C2CC2)ncc1Br.SCC 98580,c1(NC(=O)OC)cccc(C(=O)NCC(C)CN(C(=O)COC(C)CC)C)c1 98581,CCCC(C)(O)C(=O)NC1CC(CC(N2CCC2CC2CC2)=O)C1 98582,N1(C(c2ccc(C(C)=O)o2)=O)CCOCC1CC(=O)NCC1(C)CCCC1O 98583,N1(C(C(C2CCCO2)NC(CCCCOC)=O)=O)CCC2(C1)CN(C)C2 98584,CC(F)(F)CCCC(=O)N1C2CCC1CN(C(c1ccc(OC(F)F)cc1)=O)C2 98585,C1(C(=O)NCCC2(CC)CCC2)CCC(n2cc(-c3csc(C)c3)nn2)C1 98586,c1(C(=O)NC2COCCN(C(C3CC4(CSC4)C3)=O)C2)ccc2ccnn2c1 98587,N1(C(=O)CNS(=O)(=O)C2CC2)CCCC(CCNC(C2(C3CCC3)CC2)=O)C1 98588,c1(C(N(C2CCN(CC)C2)C)=O)cnc(CNC(=O)C=Cc2cncs2)nc1 98589,CC(C)C(CCNC(c1cnn(CC2CC2)c1)=O)NC(=O)Cc1cn(C)nn1 98590,c1(OC)cc(OC)cc(CNC(c2n[nH]cc2Br)C)c1 98591,c1(NC(C2CC23CC(NC(C2CCC2)=O)C3)=O)ccccc1CCO 98592,N1(CC)CC(C(=O)NCC(c2ccccc2)NC(c2ncn(CC)n2)=O)NC1=O 98593,CN1CCN(C(C2(C)CC2(C)C)=O)CC1C(=O)NCc1ccc(F)cc1 98594,N1(C(C2C(C=C)OCC2)=O)CCCN(C(c2nc(C)n(C)c2C)=O)C(C)C1 98595,c1(C(N2CC(N(C(=O)C3=COCCO3)C)C(C)(C)C2)=O)ccnc2ccncc12 98596,c1(C(=O)OC)ccc(CC(=O)NC2CN(C(=O)C=Cc3cscn3)C3CC23)cn1 98597,CS(=O)(=O)c1cccc(S(=O)(=O)N2CCN(CCNC(CC(=O)O)=O)CC2)c1 98598,C1(OC)CCn2cc(C(=O)N(C)CCN(C(=O)C(C)C#N)C)nc2C1 98599,N1(C(C)C)C(C)CN(C(=NCc2ccc(Cl)c(Cl)c2)NC2CCCC2)CC1C 98600,O=C(C1CC(O)c2ccccc21)OCc1c(F)cc(O)c(Br)c1F 98601,CC(C)CC(O)C(=O)N(C(CNC(=O)CCC(=O)c1ccc(Cl)cc1)C1CC1)C 98602,N1(CC2CCC(OC)CC2)CCCC(C)C1c1cn(-c2cc(C)cc(F)c2)nn1 98603,N1(C(CS(CC)=O)=O)CCC2(CCCCN(C(C3(c4ccncc4)CC3)=O)C2)C1 98604,C(=O)(C(C)CS(C)=O)NCc1cn(C2CN(C(C=C(C)C(C)(C)C)=O)C2)nn1 98605,c1(OC)ccc(CCC(=O)NCC(C)N(C)C(c2ccc[nH]2)=O)cn1 98606,C(CC(=O)N(C(C)CNC(=O)C=C(C)C(C)C)C)N(CCC)C 98607,Cc1nc(C(=O)NCC2(CNC(C3CC34CCCC4)=O)CCC2)cn1C 98608,C1(CC)(CC)CC(NC(=O)Cn2nccc2C)CN1C(=O)CSC1CC1 98609,C(=O)(C(O)CC(F)(F)F)N1C(C(=O)NCCN(CCC)CCC)C(CC)CC1 98610,Cn1ncc2c(C(N3CCC3CNC(c3ccc4c(n3)CCO4)=O)=O)cccc12 98611,CC12CC(NC(c3csc(O)n3)=O)(C1)C1(CN(C(=O)CC3=NNC(=O)C3)C1)O2 98612,Cc1cc(CCC(c2nnnn2CC2CC2)NCc2cc(N(C)C)no2)no1 98613,C(C)(CN(C(C(=O)OC(C)(C)C)=O)CC(F)F)(CO)OC 98614,C1(COC)CCCC(N(CC(F)F)CCF)C1 98615,c1(C(=O)OC(C(=O)Nc2c(C)ccc(N(C)C)c2)C)ccc(S(=O)(=O)N(C)C)cc1 98616,C(CC(C(=O)N1CC(SC)C1)NC(=O)CC1CC=CCC1)OCC 98617,c1(NC(COc2cc(C)on2)=O)cccc(NC(=O)CC2CCNC(=O)C2)c1 98618,c1(C(=O)NCC(C)NC(=O)CN(C)C(N)=O)ccn2ncc(Br)c2n1 98619,N1(C(=O)C=CC2CCCO2)CCC2(NC(=O)C(F)(F)c3cscn3)CCCC12 98620,N1(C(CCc2ncc(C)[nH]2)=O)CCC(O)CC1C1CC1 98621,N1(C(C(CC)O)=O)CC2CCCC(CNC(c3ncccc3F)=O)(C2)C1 98622,c1(NC(C(C)C)=O)cc(CNC(=O)NCCCN(C)C)nn1C 98623,c1(-c2cc(C(=O)NC(C)C(C)NC(C3CC(O)C3)=O)no2)cccc(Cl)c1 98624,c1(OCC)cncc(C(=O)NCC(C2CCC2)NC(=O)CC2CCN(C)C2=O)c1 98625,c1(CCC(=O)NCC(CC)NC(c2cn(CC(=O)OC)nn2)=O)ncccc1C 98626,CC1CC(C(=O)NCc2occc2C(=O)NCCc2ccncc2F)CCS1 98627,c1(CC)cc(N2CC3C(CNC(c4n[nH]cc4Cl)=O)C3C2)nc(CC)n1 98628,CCC(O)CC(=O)NCC(C)(F)CNC(c1c(C)nsc1C)=O 98629,N1(C(C(N2CCC(OC)CC2)(C)C)=O)CC2CN(C(=O)C=C(C)C)CCC2(CO)C1 98630,N1(C(c2c[nH]c(=NC)s2)=O)CCC(NC(=O)CN2CCCNS2(=O)=O)C(F)C1 98631,Cc1ccn(CC(=O)NCC#CCNC(c2sc(C(C)(C)C)nc2C)=O)c(=O)c1 98632,C12CC3(CCC3)CN1C2=O.c1(C(=O)NC(C)C(=O)NC2CC2)cc(=O)cc(Cl)[nH]1 98633,CCCCS(=O)(=O)NC(C)C(=O)NC1(CCNC(c2nnn(CC)c2C)=O)CC1 98634,N1(C(C(CC)=CC)=O)CCN(C(c2ccc(Cl)c(CC)c2)=O)C2(CC2)C1 98635,C1(C(=O)NC(C2CCCCN2C(=O)CC(O)CN(C)C)C)CC(C)(C)CN1C 98636,C1(C(=O)NC2(CO)CN(C(=O)CC3OCCCO3)C2)CCC2(CCOC2)O1 98637,N1(C(c2cnc(SC)s2)=O)CC(C)CCC1CNC(=O)CN(C)S(N)(=O)=O 98638,C1(CNC(=O)C(F)Cc2ccccc2)CN(C(=O)C=Cc2cc[nH]n2)CCCO1 98639,C(CN=c1[nH]cnc(Cl)c1CO)N(C(C1Cc2ccccc2O1)=O)CC 98640,N1(C(c2c(SC)snn2)=O)CCCCC1CCCNC(C1CCS1(=O)=O)=O 98641,c1(C(=O)NCC2(C)CCCN2C(c2cccc[n+]2[O-])=O)ccc2scnc2c1 98642,C1(CNC(COCC=C)=O)COC(C(F)(F)F)CN1C(=O)CC1CCC(C)CC1 98643,CCCCCCC(C)(CC)C(=O)NCC(C1(O)CN(C(=O)C(C)(C)CC)C1)(C)C 98644,N1(C(C)=O)CC2CC(NC(=O)C(c3nnsc3C)NC(C3CCCCC3)=O)CC2C1 98645,c1(C(N2CCC(O)(C(N3CCOC(CO)C3)=O)C2)=O)c(F)cncc1F 98646,C#CCC(CC#C)C(=O)N(C)CC1(O)CCN(C(C2(C)CCN(C)CC2)=O)C1 98647,CC1CN(CC(=O)CCc2c(F)cccc2F)CC2(CCCOC2)O1 98648,CCC(O)CC(=O)N1CC(CC(C)NC(c2cc(-c3cccs3)on2)=O)C1 98649,C1(C(=O)NCCN(C(=O)CCCc2ccncc2)C2CC2)CCC2(CCC2)OC1 98650,C1(C(=O)NCC(C(C)C)NC(CC(C(F)(F)F)OC)=O)COc2ccccc2O1 98651,N1(C(c2oc(C)c(Br)c2)=O)CCN(C(c2cc(CO)on2)=O)CC1C 98652,CN1CCOC2(CN(C(=O)CC3(N(C)C(C4CC=CCC4)=O)CC3)C2)C1 98653,CC1CC(C(=O)NC2C=CCC2)N(C(C2CCOC2(C)C)=O)C1 98654,C(CC(F)F)(C(=O)NCCC1(C)CCCO1)N(C)C(C1CC(C2CC2)=NO1)=O 98655,N1(C(C2CN(C3CN(C4CC4)C3)C(=O)C2)C)CCC(C2CN(S(=O)(=O)C(F)F)C2)C1(C)C 98656,C1(c2cn(CC3CC(F)(F)C3)nn2)(NC(=O)CC2CCCO2)CCCOC1 98657,C(=O)(CCCC(C)(C)NC(=O)C=Cc1cccnc1)N1CCC(CC)C1 98658,C1(NC(c2coc(C(F)F)n2)=O)CN(C(=O)CN2CCOCC2=O)CCC1O 98659,N1(C(C2(CNC(C3CCSC(C)C3)=O)CC(=C)C2)=O)CCOC(C)(C)CC1 98660,C(=O)(C(CNC(c1csc(F)c1)=O)CC1CCCC1)N(C)CC1(CO)CCC1 98661,C1(NC(C(CC)NC(C)=O)=O)CN(C(=O)C(C)(C)COC)CC1SC.C1CNO1 98662,c1(CNC2CCCN(c3cc(CC)ncn3)C2)cc(Br)ccc1OCCC 98663,C1(N(C(=O)C=Cc2ccoc2)Cc2c(C)snc2)CCN(c2cccnc2)CC1 98664,N1(C(=O)CCCc2ccccc2)CCN(C(=O)C(O)C2CCC2)C(CF)C1 98665,N1(C(c2c(C#N)ccs2)=O)C2CC1CN(C(=O)CC1CCCC13CC3)C2 98666,O=C(CCCCCCNC(C1CCOC(=O)CC1)=O)NC1CCC=CCCC1 98667,C(CCN=c1[nH]c(N2CCN3CCOCC3C2)nc2c1SCC2)SCC(C)C 98668,CCCC(C)(CC)C(=O)NCc1ncccc1CNC(=O)Cc1ccsc1C 98669,c1(OC)ccc2c(c1)C(C)CN(C(=O)C(N1CC(=O)N3CCCC3C1)=O)CC2 98670,C1(C(N(C2CCN(C(c3cc(CCCO)on3)=O)C2)C)=O)CCCS(=O)(=O)N1 98671,C1(C(=O)NC(CC)C(=O)N(C)C)CC(NC(C2(C)CC(C)=NO2)=O)C(O)C1 98672,c1(C(N2CC(CNC(CN(C(C)C)C)=O)C(C)CC2)=O)cn2cc(Cl)cnc2n1 98673,c1(CNC(c2cc(CNC(C(CC)(C)O)=O)no2)=O)cc(C)cc(F)c1 98674,Cc1cc(C(F)F)n(CC(=O)NC(CNC(=O)C(C)CC2CCC2)C2CCC2)n1 98675,N1(C(C(=O)NCC)=O)CCOC2(CCN(C(c3cc(C)nc4c3cnn4C)=O)C2)C1 98676,CC1CN(c2nnc(-c3cc(CN(C)C)[nH]n3)n2C)CC(c2ccsc2)O1 98677,c1(CNC2CCN(C(Cc3ccc(OC(C)=O)cc3)=O)C2)c[nH]c2cccnc12 98678,CCCCCC(C)CC(=O)NCCN(C(=O)C(F)CC1CCCC1)C 98679,N1(C(c2cccc(C(C)C)n2)=O)CC(CNC(=O)COC2CC2)N2CCC1C2 98680,C(CC(F)F)(C(=O)NCc1cc(O)cc(F)c1)N(C)C(c1ccnc(CO)c1)=O 98681,C1(NC(c2ccc(COC)s2)=O)CCC(NC(=O)C(C(C)O)NC(N)=O)CC1 98682,n1(CC(=O)NC2C3N(C(c4c(C)cn(C)c4)=O)C(CC3)C2)cc2ccccc2n1 98683,N1(C(CS(CC)=O)=O)CCC2CN(C(c3cn4cccc(C)c4n3)=O)C(C)C12 98684,C1(CNC(C2N(C(N)=O)CC(O)C2)=O)CC2(CC2)CN1C(=O)CCC1CC1 98685,C1(c2n(C)ccn2)CN(C(=O)CC2CCNC2=O)CCN1C(c1cccs1)=O 98686,c1(SCCOc2ccc(-c3n(C(C)C)ncc3)cc2)ccc2ncccc2n1 98687,N1(C(=O)CC23CCCC2C3)CCN(C(c2cc(F)c(CO)c(F)c2)=O)CC(O)C1 98688,c1(C(=O)NCC2(C)CC(NC(c3c(C)cnnc3)=O)C2)nc(C2CC2)ncc1Cl 98689,N1(C(C(C=CC)O)=O)CCN(C(=O)NCCCOCc2ccccc2)CC1 98690,Cc1cc(C(N2CCCC2CCCNC(C2CC23CCSCC3)=O)=O)nc(C)c1 98691,CC(C)CC(C(=O)NC(CCF)C(=O)NCCCOC1CCC1)C(N)=O 98692,c1(C(=O)NCCN(C)C(c2ccc(C(F)C(F)(F)F)cc2)=O)ccnc(Cl)c1N 98693,c1(C(=O)NCC#CC(=O)NCC2CN(C(C)=O)C2)c[nH]c(=S)cn1 98694,c1(C(=O)NC2CN(C(CSc3n(C)ncc3)=O)C2)cncc2c1CCCC2 98695,C(=O)(NNC(=O)c1ccc(I)cc1)NCC(C)C#N 98696,Cc1c(Cl)ccc(Cl)c1NC(=O)CC1CCCN1C(=O)Cc1ccc(Br)cc1Br 98697,C(=O)(CC(C)CC(=O)NC1(CCNC(C2CCN(C(=O)OC)CC2)=O)CC1)OC 98698,c1(COC)csc(C(=O)N(CCNC(C2CCCC2O)=O)C2CC2)c1 98699,N1(C(C(CC#C)C)=O)C2CCC1CN(C(=O)Cc1ccc(Cl)nc1F)C2 98700,C12(C(N3CC(O)CC(NC(c4ccncn4)=O)C3)=O)CCCC(CCC1)C2O 98701,C(C)(CCC(F)(F)F)(C(F)(F)F)NC(CNc1ccc(OC)cc1)=O 98702,C(=O)(CCC(C)(C)F)NC(COC)CNC(=O)C(c1ccccc1)O 98703,CC1CCC(NC(c2c(C(F)F)cccc2F)=O)CN1C(c1cccc(N)n1)=O 98704,C1(C(N2C(CNC(=O)Cc3cnns3)CC2)=O)CC12CCCCCC2 98705,c1(C(N2CCC(N(C(C(C)=C3CCCC3)=O)C)C2)=O)c(C)c[nH]c1CC(N)=O 98706,C1(C#N)(C(=O)NC(Cn2cc(CNC(CN3CC(C)C3)=O)nn2)C)CC12CCC2 98707,C(=O)(CCS(C)(=O)=O)NCC(C)(CO)NC(=O)CSCCCc1ccccc1 98708,N1(C(C(CN(C)C)N(C)C)=O)CC(O)(C2(CNC(C3(C)COCCO3)=O)CC2)C1 98709,C1(CCNC(=NCCC)NC2CCNC(=O)C2)CCC2(CC1)OCCO2 98710,c1(CNC(Cn2cc(CNC(C3(C)C(C)(C)C3)=O)nn2)=O)ccncc1F 98711,c1(C(N(CC(C)N(C(=O)C(c2ccc(C(F)F)cc2)C)C)C)=O)cc(Cl)cn1C 98712,C1(CNC(Cc2c(C)nc[nH]2)=O)CN(C(=O)CC2CCC(C)C(C)C2)CCCO1 98713,Cc1nc2c([nH]1)CN(C(C1CCCCCN1C(C1COCC(C)O1)=O)=O)CC2 98714,CC(C)CC(CNC(c1cnn[nH]1)=O)C(=O)NCCc1ncon1 98715,N1(C(c2cc(CC)sn2)=O)CC(C(N2CCCC2CNC(N)=O)=O)C(C)C1 98716,c1(Cn2ccc(NC(=O)Cc3cc(O)no3)n2)cccc(F)c1[N+](=O)[O-] 98717,C1(C(N(CCCNC(C2CC(n3cnnc3)C2)=O)CC)=O)CCC(=O)NC1 98718,C1(CNC(C2(NC(C(CC3CCC3)OC)=O)CCSC2)=O)CCCCC1(C)C 98719,c1(C(=O)NCCCCN(C(Cc2cc(C)sc2C)=O)C)cc(O)nc(O)n1 98720,c1(C(=O)OC)cc(C)nc(N(C(C)CNC(=O)Cc2cc(C)ns2)C)n1 98721,C1(C(=O)NC(CCCC)C)CCC(C(C)C)N1C(=O)CCc1nncs1 98722,Cc1c(C(=O)NCC2(CNC(C3CC4C(C3)C4(C)C)=O)CCCC2)cccc1N 98723,Cc1cc(C(=O)NC2CC2NC(c2nccnc2C)=O)cc(C)c1Cl 98724,C1(NC(=O)CC2COCCO2)CCOC12CCN(c1ncc(O)cn1)CC2 98725,C(=O)(C1=C(C)S(=O)(=O)CC1)NCC1N(C(C(CC)(C)CO)=O)CCC1 98726,c1(OC)c(NC(C2CC(F)CN(C(=O)CCC3CC3)C2)=O)cccc1Cl 98727,CC1(C)Cc2c(cnn2-c2ccccc2)CN(C(c2cc(I)cs2)=O)C1 98728,C1(CCNC(CCCNC(N)=O)=O)CCN(C(=O)Cc2ccsn2)CC1 98729,O=C(C1=CCCOC1)NC1CCN(C(=O)Cc2cnc(C3CC3)[nH]2)CC1F 98730,CCCCS(=O)(=O)CC(=O)N1CC2C(CN(C(=O)Cc3cn(C)cn3)C)C2C1 98731,n1(CCC(=O)NC2CN(C(C3CC3C(F)(F)F)=O)CC2O)ncc2c1CCCC2 98732,N1(C(C=CC)=O)CCC(C(C)NC(C2(CCS(N)(=O)=O)CCC2)=O)CC1 98733,C1(NC(c2ccc(C)o2)=O)CC2CCC1CC2NC(=O)CC1C=CCCC1 98734,N1(C(C2C(NC(CNC(C3C(C)C3)=O)=O)CCO2)=O)CCC(SC(N)=O)CC1 98735,C1(CCC)CN(C(c2nc[nH]n2)=O)CCN1C(=O)Cc1ccnc(Br)c1 98736,C1(C)(C(=O)NCC(C(=O)OC)C)CN(C(=O)C(C2CCC2)OC)C(C)(C)C1 98737,N1(C(CC2C(C)CCCC2)=O)CC2CN(C(=O)CCNC(=O)CO)CC(C1)O2 98738,N1(C(C2C(C=C)C2)=O)CC2CCC1C(NC(=O)C(C)Oc1cccc(F)c1)C2 98739,C(CC(CC)CCCC)(c1n(CCOC)nnn1)NC1CC(CCOC)C1 98740,c1(C(N2CCC(CC)(NC(=O)CCCCF)CC2)=O)cccc2c1C(=O)NC2=O 98741,c1(N2CCC(CC)CC2)nc(=NCCC(F)(F)C(F)F)[nH]c2c1CCC2 98742,C=CC1CCC1C(=O)NCC1(NC(=O)Cn2ccc(C)n2)CCC1 98743,N1(C(c2scc(OC)c2)=O)CCC(C=CC(=O)NC(C)CC2CCC2)CC1 98744,C1(C(N2C(C(N(CC(C)(C)N(C)C)C)=O)COCC2)=O)CC2(C1)CC2(F)F 98745,c1(C(=O)NCC(C)NC(c2c(CC)nc[nH]2)=O)ccc(F)c(Cl)c1N 98746,N1(C(C2(C)CC(F)(F)C2)=O)CCC(O)C(NC(C2CC23CCC3)=O)C1 98747,c1(NC(CCC2(C)CC2(F)F)=O)ccnc2c1CCO2 98748,CC1(C)SCC=C1C(c1nnnn1C1CCCCCC1)NC1CSCCSC1 98749,c1(CN(C(C(=O)OC(C)(C)C)C2CCCC2)CC)cccc(C)c1F 98750,C12(CNC(C3N(CC)CC3)=O)COCCN1C(=O)CN(C(c1cnc(S)[nH]1)=O)C2 98751,c1(CC)ocnc1C(=O)NC(C)C(CO)NC(c1cc(F)n[nH]1)=O 98752,C12(NC(C(CC)CC)=O)CC3CCC(C1C2)N3C(=O)Cc1cn(C)nn1 98753,c1(N2C3CN(C(C4(CC)CCOCC4)=O)CC2CC3)ncnc2cc(C#N)ccc12 98754,N1(C(C2CC(C)C2)=O)CCC2CCCC(C1)N2C(=O)COc1ccc(F)cc1F 98755,c1(N2CCCC(C#N)C2)nc2c(c(=NC3CCc4nn[nH]c4C3)[nH]1)COC2 98756,C(=O)(C(C)(C)C(C)O)NCC1(C(C)NC(c2nc(CC)sc2)=O)CC1 98757,c1(OC)cc(OC)cc(C(=O)OCCSCc2cc(Br)oc2Br)c1 98758,C(C)(C)(CC(=O)N1CC(C)(CCC(N2CCOCC2C(C)C)=O)C1)OC 98759,N1(CC)CCOC(C(N2CCC(CNC(C3(COC)CC3)=O)C2)=O)C1 98760,Cc1cc(C(=O)NCCCNC(=O)CC2CC2C)c(C)n1-c1nccs1 98761,C1(CC(=O)N(CCCN(C(=O)CC2(O)CCC2)C)C)CCOC(C)(C)C1 98762,C1(NC(c2c(C)cc(C)s2)=O)CCN(C)C12CCCN(C(c1ccc(Cl)s1)=O)C2 98763,c1(C(c2nnnn2Cc2ccccc2)NC(C)CCF)cc(Cl)n(C)n1 98764,c1(C(N(CC(CC)NC(=O)CCCn2cncn2)C)=O)cnn2cccc(Cl)c12 98765,C1(C(N(CCOC)CCNC(c2cc(Cl)cn2CC)=O)=O)CCC2CC2CC1 98766,C1(C(N(C)Cc2ncc(C)o2)=O)CC12CC(NC(=O)CC1CCOC1C)C2 98767,c1(C(=O)OC)cc(C(N2CC(CNC(=O)CCC3CCCO3)(OC)C2)=O)nn1C 98768,n1(CCC)ncc(C(=O)NCCC2(NC(c3cc(C)cs3)=O)CCC2)c1C1CC1 98769,CC(CCN(C)C)C(=O)NC1CC(C)N(C(=O)CCC(=O)N(C)C)C1 98770,C1(CN(C(c2n(CC)nnc2)=O)C)COCCN1C(c1nncs1)=O 98771,C#CCC(CCOC)NC(=O)C(C)N(C(C1CNC(=O)C1)=O)CC 98772,C(=O)(CC(CC)NC(=O)C(O)C1CC1)NCC(=O)OCC=C 98773,C1(N(C)C(c2ccccc2F)=O)CC2CC1N(C(C1CN3CCC1CC3)=O)C2 98774,c1(CC)nc(C(=O)NC(C)C(=O)NCC2CCN(C(C)=O)C2)co1 98775,N1(C(COCCCOC)=O)CCCC(C2CCN(C(=O)COCCF)CC2)C1 98776,C=CCCCC(=O)NCC1CCCC(CNC(=O)CCc2cnc(C3CC3)o2)C1 98777,C1(C)(NC(CC2(C)CCC2)=O)CCCN(C(C2CC(C)(F)C2)=O)C1 98778,C=CC1(C(=O)NCC2(C)CCCN2C(c2cccc(CO)c2C)=O)CCOCC1 98779,c1(NCCCNS(NC)(=O)=O)cc(S(=O)(=O)N(C(C)C)CC2CC2)ccc1C#N 98780,CC#CCC(C)NC(=O)CN(CCC)C(c1cccnc1)=O 98781,C1(CNC(c2nc(CC)sc2)=O)CCC(C)N(C(c2cnc(C3CC3)o2)=O)C1 98782,C(=O)(C(CN=[N+]=[N-])NC(c1n[nH]c2c1CCC2)=O)NCC1CCCN(C)C1 98783,N1(Cc2cn(CCCNC(C(CC=C)NC(C)=O)=O)nn2)CC(O)CCC1=O 98784,CN=c1ncc(-c2ccc(CNC(C3(c4ccccc4C)CC3)=O)cc2)c[nH]1 98785,CCC1=C(C(=O)N(C)CC2CCCN(C(c3cnncc3NC)=O)C2)CCCO1 98786,N1(CCC(=O)NC23CC(C2)N(C(c2cnoc2C2CCC2)=O)C3)C(=O)CCC1=O 98787,c1(C(=O)NCCN(C(=O)CC2C(=O)NN=C2C)CC)ccc(P(C)(C)=O)s1 98788,CC1CN(C(=O)C=Cc2nccs2)CCN(C(C2CC=CC2)=O)C1 98789,c1(C(=O)NC2CCCCN(C(C3N(CC)CCC3)=O)C2)c(C)c(C)nn(C)c1=O 98790,c1(C(c2cnn(C)c2)N(CCCC)C(C2COC(CN(C)C)C2)=O)ccccc1C 98791,c1(C(N2C(C(C)NC(C3(C)CCCO3)=O)CCC2)=O)cn(C)c(=O)n(C)c1=O 98792,C(=O)(C#CC1CCOC1)NCCN(C(c1cnc(C(C)C)s1)=O)CCOCCO 98793,N1(C(C2(C)N(C)CCC2)=O)CCCC(CO)(CNC(=O)CCc2cnccn2)C1 98794,c1(CCCCC)cc(C(=O)NC2(CO)CN(C(c3cc(C(N)=O)co3)=O)C2)n[nH]1 98795,c1(CCCNC(CCC)(c2nnnn2C(C)(C)C)C2CCCO2)ccccc1Cl 98796,C1(CNC(C2(CF)CCC2)=O)CCCC1C(=O)NCc1cscn1 98797,c1(COC)ncc(C(=O)NC(C)(CNC(C2CNC(=O)N2)=O)C2CCC2)s1 98798,CC(N=c1nc(N2CCC(CCF)CC2)c2c([nH]1)CSC2)C1CCCO1 98799,N1(C(c2cc(Cl)ccn2)=O)CC2(CCCN2C(=O)N(CCCl)CCO)C1 98800,c1(NC(C(=O)NCCC2CCCS(=O)(=O)C2)=O)cccc2c1OCCC(=O)N2 98801,N1(C(C2CN(C)C(=O)C2)=O)CC2(CCCC(CNC(=O)C(F)=CCCF)O2)C1 98802,c1(C(=O)OCC)cc(-c2cn(-c3cc(Br)nn3C3CCCCO3)nn2)ccn1 98803,c1(NC2CN(C(CC(C)c3ccccc3)=O)CC2C)cccc(F)c1C#N 98804,C(=O)(CS(=O)(=O)C1CCCC1)NCC1CN(C(C(CSC)OC)=O)C2(C1)CCC2 98805,N1(C(CNC(c2ccc(Cl)cc2)=O)=O)CC2CC2(NC(C2C3CCCCC23)=O)C1 98806,C#CCC(C)(C(=O)NC1CC1(C)CCC)NC(=O)CCOC1CCCC1 98807,C1(C(N2CCCCCC2)C(=O)NC(c2ccccc2)C)C2CCOCC12 98808,C(c1c(C)cc(C)cc1C)=CC(=O)NCC1(F)CN(C(C(CCC)OCC)=O)C1 98809,c1(C(=O)NC(CC=C)CNC(C2CCCCCN2C)=O)cc2cc(C)ccc2o1 98810,C1(C)(CCNC(C2N(CC)CCC2)=O)CCN(C(=O)CCc2cccn2C)C1 98811,c1(-c2c[nH]c(=NCc3c(OC)c(F)ncc3)s2)cccc2sccc12 98812,C(CC(F)F)(C(=O)N(C12CCC(CC1)CC2)C)n1cc(-c2cccc(C)n2)nn1 98813,Cc1nc2cc(C(N3CC(NC(=O)CC(C)P(C)(C)=O)C(O)C3)=O)cc(O)c2[nH]1 98814,C1(C(=O)NCCN(C(C2(COC)CCCCO2)=O)C)CC(=O)N(OC)C1 98815,c1(SCC(=O)N(C)Cc2cc(COC)no2)cn(C)nc1SC 98816,c1(NC(C(c2cc(CC)on2)N(C(C)CCC#N)C)=O)cccc(OC)c1 98817,c1(C(=O)NCC(CNC(CCCNC(N)=O)=O)F)sc([N+](=O)[O-])cc1Cl 98818,c1(C(N(c2c(O)nc(=O)n(Cc3ccco3)c2N)CC)=O)ccn2nccc2c1 98819,C(C(C(=O)NC(C(=O)N(C)Cc1ccn(C)n1)C1CCCC1)OC)OC 98820,c1(C(=O)NC2C(NC(CC(C(=O)OC)C)=O)CCOC2)cnc2[nH]nnc2c1 98821,c1(NC(c2cccc(Br)c2)=O)ccc2[nH]cc(-c3ccc(C(=O)O)c(F)c3)c2c1 98822,c1(C(N(CCCOCCN(C(C(C)SC)=O)C)C)=O)c(C)oc2ccccc12 98823,CC(CCCc1ccccc1)C(=O)NC1(CNC(c2cnco2)=O)CCOC1 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98858,C1(C(=O)Nc2ccc(C)cc2S(=O)(=O)NCCSC)CC(C)c2ccccc2N1 98859,N#Cc1cnc(N2CCC(F)(F)C(CNC(c3cccc(Cl)c3Cl)=O)C2)c(Cl)c1 98860,N1(C(c2sc(C)c(Br)c2)=O)CCC2CN(C(c3c(F)cccc3Br)=O)CC12 98861,C1(CNC(C(C)(C)OCC)=O)(OC)CCN(C(C2COCC(C)O2)=O)C1 98862,Cc1cn2ccnc(C(=O)NC3CCCC3CNC(c3cn(C)nn3)=O)c2n1 98863,CC(=O)CCCCC(=O)NCC(CNC(=O)C(c1ccnn1C)C)CO 98864,CONC(=O)C(=O)NCCC1CCC(NC(C2C3CCCCC23)=O)C1 98865,C1(C(N(CCC(C)NC(=O)Cn2cnc(C(N)=O)n2)C)=O)C(C)(C)C1(F)F 98866,c1(CC)cc(C(N2CCCC(NCc3ccc(CBr)cc3)CC2)=O)ccc1O 98867,C(=O)(CN1C(=O)Cc2ccccc21)NC1CCCC(OC2C(=O)NCC2)CC1 98868,C1(NC(c2c(OC)cccc2)=O)COC2(CCN(C(c3coc(CO)c3)=O)C2)C1 98869,c1(CN2CC(OC)C(NC(=O)C(C)(C)NC(C)=O)CC2)c[nH]c2cc(Br)ccc12 98870,c1(CC(N2CCC(NC(Cc3c(C)cccn3)=O)C2)=O)ccc2oc(O)nc2c1 98871,C1(CC(=O)NC(CC2CN(C(C(C)OC)=O)C2)C)CCC(C(F)(F)F)O1 98872,N1(C(C(C(C)C)C)=O)CCC2(CCCC2NC(=O)C=CC2COC(C)(C)O2)CC1 98873,C1(C(=O)NCc2c(C)nccc2)CCC(O)CN1C(c1cccc(F)c1O)=O 98874,c1(NC(=O)NC)cccc(C(=O)NCC(C)(C)NC(C2CCC(O)C2)=O)c1 98875,C1(C(N(C2CCCCC2O)C)=O)(CO)CCN(C(C2CCC(C(N)=O)C2)=O)C1 98876,C12(NC(=O)CCC3CCCO3)CC3CCC(C1C2)N3C(=O)CC1(C(F)(F)F)CC1 98877,N1(C(C2(OCC)CCSCC2)=O)CCCC(NC(=O)CC2(C)CC2(F)F)CC1 98878,c1(C(=O)NCCOC2CN(C(c3cc(C(N)=O)[nH]n3)=O)C2)noc2c1CCCC2 98879,c1(CNC(=NCCOCC=C)NCC2CCC(CO)O2)cccc2c1NCCC2 98880,c1(C(=O)NC2CCC(NC(C(CC)OCC)=O)C2)ccc(OC)cc1F 98881,C(=O)(CC(C)CC(C)(C)C)NC(CCNC(c1c(C)ncs1)=O)C(C)C 98882,c1(C(C(=O)C(F)CC2CCC2)=O)cc(OC(F)F)cc(F)c1.C(CNC1CC1)N 98883,n1(CC(N2CC(O)CC23CCOCC3)=O)ncc2c(Br)cccc2c1=O 98884,C1(C(=O)NCc2n(CC)ncn2)CC2CC1CC2NC(c1cc(C)nnc1C)=O 98885,C1(C2CCN(C(C3CCCOCC3)=O)CC2)(NC(C(C(C)C)NC(C)=O)=O)CC1 98886,C(=O)(C(C)C(=O)NC1(CO)CN(C(C2(CO)CCC2)=O)C1)OC 98887,C(=O)(C1c2c[nH]nc2CN1C(=O)CCNC(C)=O)NCCOCCC 98888,C1(CNC(CC2CCCN(C)C2)=O)CN(C(=O)Cc2cccnc2)C(C)(C)C1 98889,c1(C(N(CCC)CCNC(C2(F)CCC2)=O)=O)cc(C)c2c(c1)CCC2 98890,C1(CC)CN(C(c2cnns2)=O)CC1NC(c1ccc(C(C)(C)CC)cc1)=O 98891,CC1C(=O)Nc2ccccc2N1C(C1CC1c1ccccc1OC(F)F)=O 98892,C#Cc1cnn(C)c1C(N1CCC(C(C)NC(=O)C(CCC)OCC)CC1)=O 98893,c1(SC)cccc(C(N2CCC(NC(c3cncc(C)n3)=O)C2)=O)c1O 98894,N1(C(c2ccc(SC)o2)=O)CCC2(COC(CNC(C3(C)CCSCC3)=O)C2)C1 98895,c1(C(=O)NC(CN(C(c2cc(CCC)n(C)n2)=O)C)C)c[nH]cc(Br)c1=N 98896,c1(C(N(CCNC(C2CCC(COC)O2)=O)CC)=O)c(Cl)ccc(OC)c1N 98897,c1(CN2CC(F)CC(C(N3CC(CC)OCC3)=O)C2)c(Cl)ccc(Br)c1F 98898,C1(CNC(c2ccc(I)c(O)c2)=O)CCNCC1(F)F 98899,C1(C(C(=O)NCCOCC=C)C)CCNCC1 98900,C(=O)(C1=C(C)CCOC1)N1CC2C(CC(=O)NC(C#CC)(C)C)(CC2)C1 98901,c1(C(N2CC(CCNC(C3CC(C)(CC)C3)=O)C2)=O)cc(C)ccc1[N+](=O)[O-] 98902,CC(C)C(F)(F)CC(=O)NC1CCC(C)N(C(c2cc(=O)c(Br)c[nH]2)=O)C1 98903,C1(CC(=O)NCCC(CNC(C2OCCC2C(C)C)=O)OC)CCCN(C)C1 98904,c1(C(=O)NCCN(C(=O)CNC(c2ccc(Cl)s2)=O)C)cc(C(F)F)nn1C 98905,c1(CC(=O)NCC(C)NC(C(CCCC)O)=O)coc2c(Cl)c(Cl)ccc12 98906,C1(NCCC(COC)(C)C)C(C)N(C)CCN1C 98907,c1(CC)cccc(C(=O)NC2CCC2CNC(C2(C)C=CCC2)=O)c1N 98908,c1(NC(CN(C(COCCCC#C)=O)C)=O)ccc(C)cc1.C1(=O)CCN1 98909,C1(NC(c2ccc(CSC)o2)=O)COC2(CCN(C(c3cc[nH]c3)=O)C2)C1 98910,c1(CC)cc(C(=O)NCCCN(C(=O)CCc2cccnc2F)C)cn(C)c1=O 98911,c1(C(N2CC(C)OC(CO)C2)=O)ccc(S(=O)(=O)N(C)C)cc1.C1C(=O)N1 98912,N1(C(Cc2cc(C)c(Br)cc2)=O)CC2CCN(C)C2C1 98913,C(S(=O)(=O)C(C)C(=O)N(c1cccc(C)c1)C1CC1)c1n(CC)ncc1 98914,Cc1c(C(N2CC3C(N(C(=O)C(F)CC4CC4)C)C3C2)=O)oc2c(Cl)cccc12 98915,c1(C(=O)NC(COC)CNC(=O)CCc2conc2C)cc(F)ccc1N 98916,c1(C(C)=O)cc(=NCC2CN(C(C3CC(C)CO3)=O)CCO2)[nH]cn1 98917,N1(C(C2CC=C(C)CC2)=O)CCCC(C2CC2NC(=O)C(C)(C)C(F)F)C1 98918,CC1C(=O)N(C)CN1C(=O)NC1CCn2ncnc2C1 98919,c1(C(CSCCOC)O)cccc([N+](=O)[O-])c1 98920,C12(C(C)C)CCC(NC(=O)C(Cn3cccn3)NC(=O)CN3CC=CC3)C1C2 98921,c1(C(N2C3CC(CNC(=O)CC4CSCCS4)C2CC3)=O)ccc2nn[nH]c2c1 98922,C(C)(C)(CC(F)C(=O)NC(C1CCOC1)CO)NC(CC1CCN(C)C1=O)=O 98923,c1(C(N2CC3C(CNC(C(C)CC(F)F)=O)C3C2)=O)nnc2ccccc2c1N 98924,CN=c1[nH]cc(C(N2CCCC(NC(=O)C(C)CSc3ccc(F)cc3)C2)=O)s1 98925,C1(CNC(C2CC3CC3C2)=O)COCCN(C(c2ccncc2F)=O)C1 98926,Cc1cc(C(N2CC(N(C)C(c3cnoc3C)=O)C3(CC3)C2)=O)nc(N(C)C)n1 98927,C1(S(C)(=O)=O)(C(=O)NC2CC(C)(NC(CC3C(C)C3(F)F)=O)C2)CC1 98928,N1(C(Cc2c(C)ocn2)=O)CCC(C)(C)C1C(=O)NCCCN1CCC(O)C1 98929,c1(CC)cn2c(n1)CC(C(=O)NCCCNC(c1ccc(C(F)(F)F)o1)=O)CC2 98930,c1(N(C)C)ccnc(C(=O)NCCC2CCCN2C(=O)C=Cc2ccco2)c1 98931,C1(NC(=O)CC2CC=CC2)CCC(O)CN(C(C2(c3ccc(Cl)cc3F)CC2)=O)C1 98932,c1(CSCC)ccc(C(=O)NC2CC(CNC(C3C(C)C3(F)F)=O)C(O)C2)cc1 98933,c1(C(N2CCC(OCCNC(COC)=O)C2)=O)cccc2nsnc12 98934,Cc1cc(-c2cncc(F)c2C(=O)Nc2cnn(CCO)c2)ccc1OC(F)(F)F 98935,N1(C(C(Cc2cccc(OC)c2)N)=O)CC(C)(C)CCC1CC(=O)O 98936,C1(CNC(c2c(C)snn2)=O)CCN(C(c2cnn3ccn(C)c23)=O)CC1(F)F 98937,Cc1sc(C(=O)Nc2ccc(-n3ccnc3)cc2)c(C)c1Br 98938,c1(C(N(C(=O)CCN2CCCC(C(N)=O)C2)C(C)(C)CSC)=O)ccc(F)cc1C 98939,C(C(C(=O)N1CCC(CN(C)C)C1)n1cc(-c2csnn2)nn1)OCC 98940,N1(C(C=Cc2c(C)ncs2)=O)CCCN(C(c2ccc(F)c(N)c2)=O)CC1C 98941,C(=O)(CCCCNC(N)=O)NC(CN(CC(=O)N(c1ccccc1)C)C)C 98942,C1(C)(C(C)(C)C)CC(C(=O)NCC(O)CNC(C2CSCCS2)=O)C1 98943,C1(NC(=O)C(O)C2CCCC2)CCC2CN(C(c3cc4c(s3)CCC4)=O)CC2C1 98944,C1(CCC#C)CCCN(C(=O)CCC(C)NC(=O)C(C)C(C)C)C1 98945,Cc1c(C(=O)NCCCCNC(c2csc(C)c2C)=O)cc(F)cc1Br 98946,N1(C(C(C)OCC(C)C)=O)CC(NC(=O)CCc2nc(O)n[nH]2)C(C(F)(F)F)C1 98947,C1(COC)CCCC1NC(=O)CC1(C)CCN1C(C)=O 98948,CCC(CC(=O)NC1CCC12CN(C(c1cc[nH]n1)=O)C2)C(C)C 98949,c1(-c2onc(CN(C(=O)OC(C)(C)C)CC)n2)cc(CO)cc(C)c1 98950,C1(CNC(c2c(C(C)C)csc2)=O)CCCCN(C(=O)COc2ccsn2)C1 98951,C(C(C)CC(C)C)NC(c1ccncc1)CC 98952,N1(c2cc(NCC3(CO)CC=CC3)nc(C)n2)CCC(C)C2(CCC2)C1 98953,C1(C)(CNC(c2[nH]cc(C)c2)=O)CN(C(=O)CCNc2ccccn2)CCO1 98954,C1(NC(c2c(C)n(C)nc2)=O)CC12CCN(C(C1CC3CC3C1)=O)CC2 98955,n1(CC)nc(C)c(C(=O)NCC2(NC(=O)C(C)S(C)(=O)=O)CCCCC2)c1C 98956,C1(C)(C(=O)Nc2c(CC)noc2)CCCN1C(=O)CCCn1ccnn1 98957,c1(OC)cc(C(=O)NC2CCCC2CNC(C2(CO)CCCC2O)=O)cnc1C 98958,C1(CNC(c2cc(OC)no2)=O)N(C(=O)Cc2cc(C)cc(F)c2)CCC1(C)C 98959,N1(C(C=NOC)=O)CC(F)CC1C(=O)NCc1cnc(S)nc1 98960,c1(OC)ncccc1C(=O)NCC(C)(C1CC1)NC(c1ccoc1Cl)=O 98961,CCCCCC(O)CC(=O)NCCN(C(=O)CC(C)C)Cc1ccccc1 98962,c1(CC(=O)OCCOCCCC#C)coc2cc(F)ccc12.C(C=C)O 98963,C12(CO)COCC(Nc3ncc(Br)cc3C(F)(F)F)(C1)C2 98964,C(=O)(C(C(C)C)n1ccnc1)NC1(C)CC(NC(C2(CC)CCCC2)=O)C1 98965,c1(CN(C(C(CC)SC)=O)C)cnn2c1CN(c1nnc(C3CC3)o1)CC2 98966,Cc1ccc(NC(=O)C(=O)N(CC(C)CNC(=O)CNS(N)(=O)=O)C)cc1 98967,C1(N(C)C(c2ccsc2)=O)CN(C(=O)CN2CCCCCC2=O)CC1(C)C 98968,N1(C(CCC)=O)CCCC(C(N2CCCC2c2cc(Br)cs2)=O)C1 98969,S(=O)(=O)(c1c(C)n[nH]c1C)N(Cc1c(OCC)ccc(C)c1)Cc1cccs1 98970,c1(NC(C2CC3(CCN(C(=O)CCC4CC4)CC3)C2)=O)cc2c(Cl)cccc2s1 98971,c1(C(C)C)nc(NC(c2cccnc2N)C)cc(N2CCOCC(CO)C2)n1 98972,N1(C(=O)C2=CCCCC2)CC2OCCN(C(C3CCOC3=O)=O)C2C1 98973,N1(C(CCC=C(C)C)=O)CC(N=[N+]=[N-])CC1C(=O)NCCN1CC=CCC1 98974,C(=O)(CCC1=NNC(=O)CC1)NC1CN(C(CN(CCC)C)=O)C2(C1)CCOC2 98975,CC(C)(C)C(O)C(=O)NC1CN(C(C23CCC(C2)C3)=O)CC12CC2 98976,N1(C(C(=O)NC(C(=O)NCC(=C)C)C2CC2)C)CCOCC1 98977,C1(CC#C)(C(=O)N(CC(C)CNC(C2(COC)CCOCC2)=O)C)CCCOC1 98978,N1(C(C2(c3cc(C)on3)CC2)=O)CCC2(CC(NCc3ccc(Cl)cc3)CO2)C1 98979,C(=O)(CCCCSC)NC(C1CN(C(c2ccc(COC)o2)=O)C1)C 98980,c1(CN2C(c3ccc(C(C)C)cc3)CCOCC2)cccc(S(F)(F)(F)(F)F)c1 98981,CCCC(CCC)=CC(=O)N(C(CNC(=O)C(C)(C)n1cnnn1)CC)C 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99246,Cc1cc(C(=O)NCC2CN(C(C3CN(S(N)(=O)=O)C3)=O)CC2(C)C)ccc1Cl 99247,C1(OC)CCC12CC(C(N1CC(N3CCN(C(=O)C(C)(C)C(C)O)CC3)C1)=O)C2 99248,N1(C(C=C(CC)CC)=O)CCCCC1C1(NC(c2ccc(COC)cc2)=O)CC1 99249,C(CCC(C)(C)C(=O)N1CC2CCCC2C1)NC(CC1CCCC(C)C1)=O 99250,c1(OC)ncccc1C(=O)N(C)CC1(NC(C2CCOC2C)=O)CC1 99251,C1(O)(C(CNC(CC(=O)NCC#C)=O)C)CCN(C(=O)C(C=C)CC)C1 99252,Cc1ncc(C(=O)NCCCCN(CCCNC(=O)CCn2ccnn2)C)n1C 99253,c1(C(=O)NC2CCCC(C(=O)Nc3cc(C(C)C)no3)C2)ccc(O)cc1Cl 99254,C1(C(=O)NC2(CO)CN(C(C=C(C)CN3CCCC3)=O)C2)CCn2ccnc2C1 99255,c1(Cc2ccc(C)c(F)c2)nc(=NC(=O)N(CC(C)C)CCO)[nH]s1 99256,N1(C(CSCCN(C)C)=O)CC2(CNC(=O)CC3CNC(=O)C3)CCC1CC2 99257,c1(C(=O)NCCCN2CCC(NC(C34CC(OC)C3C4)=O)C2)cc(F)cc(F)c1 99258,Cc1nnc2n1CC(C(N1CCC(CCNC(c3cc(F)ccc3O)=O)C1)=O)C2 99259,N1(C(C2(CC)CCCCC2)=O)CCC2(C1)CN(C(c1cccc(F)n1)=O)CCO2 99260,c1(CNC(=O)Nc2c(C)ccc(C#C)c2)cc(Cl)cc([N+](=O)[O-])c1O 99261,c1(C(=O)NCCCN(C)C(C2(C(F)F)CC2)=O)cnc(Br)s1 99262,N1(C(c2c(CC)cccc2)=O)CC2(CCN(C(c3cnn(C)c3N)=O)C2)C1 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99453,N1(C(C(CN(CC)CC)F)=O)CCC(C)(CCNC(=O)Cc2cn[nH]c2)C1 99454,C1(NC(CC(c2c(C)cccc2)C)=O)COCCN(C(=O)CN2CSCC2=O)C1 99455,C(C)(CC(C)NC(C1(C(C)(F)F)CCC1)=O)NC(CCOCC#C)=O 99456,C1(CCNC(=O)Cc2cscn2)CCCN(C(C23CCCC2CCC3)=O)CC1 99457,C(=O)(C1CCc2c[nH]nc21)N(C(C1(C)N=C(C)SC1)=O)C1CC1.c12cn(nn1)CCO2 99458,N1(C(CCOCC#C)=O)CCCC(CN(C)C(C2(N3CCCCC3=O)CC2)=O)C1 99459,c1(C(N(C)CC2(O)CCN(C(C3(C(N)=O)CCC3)=O)C2)=O)cnn2c1OCC(F)C2 99460,c1(C(=O)NC2CCC2NC(C2CCCOC2)=O)ccc2c(n1)CCCN2 99461,C1(O)(CCNC(c2c(C)ncs2)=O)CCCN(C(C2CCN2C2CCCC2)=O)C1 99462,N1(C(C2CC2CF)=O)CCN(C2CCN(C(=O)Cc3cc(C4CC4)on3)C2)CC1 99463,CCC(C)CCC(=O)N1CC(O)(CCNC(C2CCC(F)CC2)=O)C1 99464,N1(CCCCNC(C(c2nc(CC)[nH]n2)N(C)CC)=O)CCCC(C(N)=O)C1 99465,C1(NC(CCCC)=O)CN(C(=O)C(=O)Nc2ccc(C)c(C)c2)CC2(CCC2)C1 99466,Cc1cc(C(N2CCCC2CCCNC(=O)C(=Cc2cscn2)F)=O)ccn1 99467,Cc1cnc(-c2cn(C3CC(NC(C4CCCN4C4CCCC4)=O)C3)nn2)nc1 99468,C(CCC(N)=O)(C(=O)NCCCN(C)C1CC1)n1cc(COC)nn1 99469,c1(N(CCCOCC)C)ncc(S(=O)(=O)N2CCC(c3ccco3)C2)cc1Cl 99470,N1(C(C(C)(C(C)C)NC(C)=O)=O)CC2CCCC(NC(c3cccn3C)=O)C2C1 99471,c1(OC)ccc(C(O)CC(=O)NC(C2CCC(=O)N2)c2nn[nH]n2)cc1OC 99472,CC1(C)CC(C)(C(=O)NC(CCOCCO)C(=O)NCCc2ccccc2O)C1 99473,n1(CC(N2CC3C(N(C(CN(CC)CC)=O)C)C3C2)=O)nc(C)ccc1=O 99474,c1(C(=O)NC2CN(C(CC(=C=C)C)=O)C3C2C3)ccc(O)cc1C 99475,C1(NC(C2CC3CC3C2)=O)CN(C(C2CCCC2)=O)CC2(CCC2)C1 99476,CC1(CNC(c2ccc(F)s2)=O)CCCN1C(=O)C(F)CC1CCCC1 99477,N1(C(C(=O)NC(C(C)C)C)=O)CCCC(C(=O)CN2CCCC2)C1 99478,C1(NC(c2nc(CC)oc2)=O)CN(C(=O)C(C)N2CC(C)C2)CCC1CO 99479,c1(C(=O)NC(C(C(C)C)NC(c2c(C)nncc2)=O)C)cc2ccc(F)cc2o1 99480,C(=O)(C(C)(CC)CO)N(CCC)CCNC(c1onc(Br)c1C)=O 99481,N1(C(CN(C(=O)CC2CCCOCC2)CC)=O)CCC(C)(C#N)C1 99482,c1(CC(=O)N(C(CCNC(CN2CC(CC)C2)=O)C)C)sc(C)nc1C 99483,C1(CNC(C2N(C)CCC2)=O)CN(C(=O)CCC2CC2(F)F)CC(C)(C)O1 99484,Cc1cn(-c2ccc(F)cc2)nc1C(=O)N(CCS(C)=O)C(C)(C)C 99485,CC1CN(C(=O)CCc2nncn2C)CCCN1C(C12CCCCC(F)(C1)C2)=O 99486,N1(c2n(CCOC)c(C(c3ccncc3)C)nn2)CC2CC(O)CC2C1 99487,C1(C2CCCN(C(=O)C(O)CCSC)C2)(NC(c2ccc(OC)cc2Cl)=O)CC1 99488,c1(C(N2C(CCCNC(CC=C)=O)CCC2)=O)ccc(-c2cn[nH]c2)cc1 99489,Cc1sccc1C(c1cnn(C)c1)NC(=O)NC1COCC1C(N)=O 99490,CC(N=c1nc2sccc2c(NCc2csc(Br)n2)[nH]1)c1cnccn1 99491,CC(CC(=O)N1CCCC(O)(CN=c2[nH]nc(CO)s2)C1)CC(C)(C)C 99492,c1(SC)cc(=NC(=O)C2N(C(=O)Cn3ccnc3)CCCC2(C)C)[nH]n1C 99493,Cc1c(C(N2CCC(C(=O)NCC(C)(O)CO)(CO)C2)=O)ncn1C 99494,C1(C(C)(C)C)CCN(C(=O)CCN(C(=O)CC2CCOC2)CCO)C1 99495,c1(CC(=O)N(CCC(C)NC(=O)C(C2CCOCC2)N(C)C)C)c[nH]ccc1=O 99496,C1(NC(C(C)CC2CCC2)=O)COCCN(C(=O)Cc2cnccn2)C1 99497,c1(C(=O)NCC(C(C)C)(C)NC(C2CCC2(C)C)=O)cc2n(c1)CCOC2 99498,Cc1c(-n2cc(C3(C)CCCN3C(=O)Cc3ccoc3)nn2)cccc1Br 99499,C(=O)(CCCC(=O)N1CCN(C(=O)CCOC2CCOCC2)C(C(F)F)C1)OC 99500,Cc1cnc(NCCc2ccc3ccsc3c2)c(S(=O)(=O)NCC2CCC2)c1 99501,C1(NC(=O)CN2CCCS2(=O)=O)CN(C(c2ccc(C3CC3)o2)=O)CC2(CC2)C1 99502,Cn1c(C(=O)NCC2(C(N3CC(N4CCOC4=O)C3)=O)CCCO2)cnc1Cl 99503,N1(C(C2C(C=C)CC2)=O)CCOCC1CNC(c1nc(Br)sc1C1CC1)=O 99504,C1(NC(C2N(CC)CC2)=O)C=CC(C(=O)N(CCC(O)CO)C)C1 99505,C(CN=c1cc[nH]cc1S(=O)(=O)N1CCC(C(C)C)C1)c1c(C)cccc1 99506,Cc1ccc(F)c(C(N2CC=CC(NC(=O)CC(C)C3CC3)C2)=O)n1 99507,c1(-n2cc(C(C)(C)NC(c3cnco3)=O)nn2)cccc(F)n1 99508,Cc1[nH]nc2ccc(C(=O)NCC(CO)NC(=O)CCCn3ccnc3C)cc12 99509,N#CC1CCN(CC(=O)NC2CC(n3cc(C4CCCC(O)C4)nn3)C2)CC1 99510,c1(CC)cscc1C(=O)NCCCN(C(c1ccncc1)=O)CC1CCCC1 99511,N1(C(CCCCC)=O)CC2(C1)CN(C(c1ccc(C3CCCO3)nn1)=O)C2 99512,Cc1ccc2[nH]nc(CNC(=O)NCCCN3CCCC(C)C3)c2c1 99513,C(=O)(C(F)C1=CCCCC1)N(CC(C)NC(c1c(C)nc(CO)s1)=O)C 99514,Cc1cccn2nc(C(=O)NCC(O)CNC(=O)C(C)Cc3ccncc3)cc12 99515,c1(NC(=O)OCC(N2CC(N(C(c3cc(OC)n[nH]3)=O)C)C2)=O)cc(C)cc(C)c1 99516,C(=O)(C(C)(C)CS(N)(=O)=O)NCC(CC)(CC)NC(c1cc2ccccc2s1)=O 99517,n1(C(C)C)ncc(C(=O)NCC(C(C)(C)C)NC(C2(Cl)CC2(F)F)=O)c1C1CC1 99518,c1(C(N2CCC(F)(CNC(c3c(CC)c(C)sc3)=O)C2)=O)ccc2c(c1)CCO2 99519,N1(C(CC2(CSC)CC2)=O)CCC(NC(=O)COC2CCCCCC2)CC1C 99520,N1(C(C2(CC)CCCC2O)=O)CC=C(C(=O)NCC2(CC3CC3)CC2)CC1 99521,C12CCC(C1)CNC2=O.c1(CCC(=O)NCC2(CC(=O)OC)CC2)cncn1C 99522,C(=O)(C(C(C)CCC=C(C)C)N1CCC(C(=O)OC)CC1)NCCCOC 99523,c1(NC)cc(C(N2CC(C)(NC(=O)C(CC3CCC3)NC(C)=O)C2)=O)cc(Cl)n1 99524,C#Cc1cccc(CNC2CC=CC(C(=O)Nc3cnc(C(=O)O)nc3C)C2)c1 99525,c1(C(=O)NC(CNC(C(C)c2cccs2)=O)C(C)(C)C)cc2occc2[nH]1 99526,CCS(=O)(=O)CC(=O)NCC1CCCCN1C(C1CCCN(C(N)=O)C1)=O 99527,C1(NC(c2c(CC)[nH]nc2Cl)=O)COCCN(C(=O)COC2COC2)C1 99528,c1(C(=O)NC(C2CCN(C(=O)C(C)Cc3ccco3)C2)C)ccnc(Br)c1F 99529,c1(C(=O)NCCCCCNC(c2c(C)oc(Br)c2)=O)ccc2cc[nH]c2c1 99530,Cc1c(C(=O)N(C)CCN2CCN(C(c3ccc(Cl)cn3)=O)CC2)cnn1C 99531,c1(C(N(CC(CNC(C2CC(CC(=O)OC)C2)=O)O)C)=O)c[nH]nc1C(F)(F)F 99532,C1(NC(CCOC(C)C)=O)CCCC(NC(=O)CCN2CCCCC2)C1 99533,c1(C(=O)NCC(O)CNC(C2CCC=CO2)=O)ccc(=NCC2CC2)[nH]c1 99534,C1(C(=O)NC(CNC(CCc2onc(C(C)C)n2)=O)(C)CO)CCN(C)C1C 99535,C1(NC(c2c(C)snc2)=O)CCCCCC1C(=O)N(C1CCCC1(F)F)C 99536,c1(CCC)cc(C(=O)NCCC(C)N(C(=O)C(C)Cc2ccncc2)C)n[nH]1 99537,C#CC1(C(N2CCCC(CCNC(C3COCCN3C)=O)C2)=O)CCCC1 99538,CCC1=NOC(C(=O)NCCC(C)NC(c2cc(C(N)=O)no2)=O)C1 99539,C1(CC(=O)NCCn2cc(CCSCC)nn2)C(=O)N(C)N=C1C 99540,Cc1cc(C(N2CC(NC(c3nc(O)c(C)s3)=O)C3CC23)=O)n2nc(C)cc2n1 99541,N#CCC(=O)NNC(=O)Cc1cc(Cl)ccc1Cl 99542,c1(OC(C)=O)ccc(C(=O)NC(C2(CN(C)C)CC2)=O)cc1.N12CCCC1C2=O 99543,C1(NC(C(C(=C)Cl)(C)C)=O)CCC2CCN(C(=O)CCNC(=O)OCC)C1C2 99544,C1(C)(CNC(C2C(c3c(C)ccnc3)C2)=O)CCC(NC(c2cc[nH]n2)=O)CC1 99545,c1(C(=O)NC(CC)(C)CNC(=O)C(C)NC(c2cccs2)=O)sc(CO)nc1C 99546,C1(C(N2CC(OCC)C2)=O)CC12CCN(C(c1cccc(F)c1F)=O)C2 99547,N1(C(CC2C(NC(CC(=O)NCC#C)=O)CC2O)=O)CCC(F)(CO)CC1 99548,Nc1cccc(C(=O)NCCOC2CCN(C(=O)C(O)CN3CC=CC3)CC2)n1 99549,C(=O)(C1Cc2ccccc21)N1CCC(C(N(CC(C)CO)C)=O)CC1(C)C 99550,c1(OC)ccc(COCCCC(=O)NC2CC(C)N(C(=O)CC#N)C2)cc1 99551,c1(C(=O)NC(C)CCCNC(C2COCCO2)=O)cnc2cc(Br)ccc2c1 99552,CC(C)(C)CC(=O)N1CCCC1C(N1CC(NC(C23CC(F)(C2)C3)=O)C1)=O 99553,N1(C(c2ccc(C(=O)OC)cc2)=O)CC(N(C)C(c2conc2C)=O)C2(CC2)C1 99554,N1(C(Cc2cccc(COC)c2)=O)CCN(C(c2nc(O)sc2C)=O)C2CC12 99555,N1(C(CC(C)CC2CCCN2C(=O)OC(C)(C)C)=O)CCCCC1C1CC1 99556,c1(C(=O)NC2CC(CNC(CN3C(C)CC3)=O)C2)cc(F)ccc1N1CCOCC1 99557,Cc1cccc(C2=CCN(C(=O)NCCC3CNCCCO3)CC2)c1 99558,C(CN=c1nc(O)c(Cl)c[nH]1)NCc1ccc(Cl)c(Cl)c1 99559,N1(C(C2N(C)CC(O)CC2)=O)CCC(C(N2CC3(CO)CC3(CO)C2)=O)CC1(C)C 99560,CC1COc2c(C(=O)N(C3CCCN(C(=O)C#CC4CCC4)CC3)C)cccc21 99561,c1(C(N2CCCN(C(CC(C)C3CCCO3)=O)CC2)=O)ncccc1N=[N+]=[N-] 99562,C(CC(=O)N1CCCC(CNC(=O)CN(C(=O)C(C)C)C)CC1)(C(C)C)OCC 99563,C(=O)(C1=C(Cl)CCOC1)NCC12CN(C(c3c(OC)cccn3)=O)C(C1)CO2 99564,C1(CNC(C=CCC)=O)CCCC(CNC(=O)C(F)(F)c2cscn2)C1 99565,c1(C(N(C(CNC(c2cc(CC)[nH]n2)=O)C)C)=O)cc(OC)c(OC)cc1O 99566,N(C(=NCCN1CCOCC1)NC(c1ccccc1F)C)CC(=C)C 99567,c1(C(N2CCN(C(C3C(C)CCCC3)=O)CC2)=O)cc(P(C)(C)=O)ccn1 99568,CCC(CC(F)F)C(=O)N1CCCC1C(=O)NC1(c2ccc(F)cc2)CC1 99569,CS(=O)(=O)CC(F)(F)CCNC(=O)Nc1nn[nH]c1C(F)(F)F 99570,N1(C(C2CC(C#C)(O)C2)=O)CCC(C)(C)C1CNC(c1cn(CCC)nc1C)=O 99571,c1(C(N2CCC(NC(C3CCCS3)=O)C2)=O)cc(F)c2cc[nH]c2c1 99572,N1(C(c2c(C)cnnc2)=O)CC(NC(c2cc(-c3ccoc3)[nH]n2)=O)CCC1C 99573,c1(COC)nn(C)cc1C(=O)N(CCNC(c1cc[nH]c(=N)c1)=O)CC1CC1 99574,N1(CCC(=O)N(C2CCN(C(C(CC)(C)O)=O)C2)CCO)C(=O)NC(C)(C)C1=O 99575,C(=O)(C1=CC2(CCOC2)C1)N(CC(C)(C)NC(=O)CCc1ccoc1)C 99576,CC(C)(CCCCNC(C1CC(C2CC2)=NO1)=O)NC(C1CC2CCC(C1)S2)=O 99577,CC(C)CC(C)C(=O)NCC1CC2CCC1N2C(C1CC=CCC1)=O 99578,S(=O)(=O)(c1ccc(Br)cc1NCC1CCCCCCC1)N1C2CC(=C)CC1CC2 99579,C1(NC(CCSC)=O)COCC1NC(C1CN(C2CCOC2)C1)=O 99580,N1(C(C(CCC#C)O)=O)CCCN(C(c2cccc(Cl)c2C)=O)C(C(C)C)C1 99581,CC(C)(O)C(F)CNC(C1(C2CCCN2C(=O)CC2CCCO2)CC1)=O 99582,CC1CC(CNC(C2COC(CNC(C3Cc4nccn4C3)=O)C2)=O)CC(C)C1 99583,CC1C(NC(c2cnccc2Cl)=O)C(C)CCN1C(c1cc(N(C)C)ccn1)=O 99584,c1(OC)ccc2c(c1)C(NC(=O)NCCc1ccc(NC(C)=O)cc1)CCN2 99585,N1(OC(C)CNC(=O)CNC(=O)C(C)Nc2ccccn2)CCCCS1(=O)=O 99586,c1(C(=O)NCC2CCCN2C(c2cnn(C3CCOC3)n2)=O)cnn2c1CCC2 99587,c1(C(=O)NC2C(NC(C3CC(C)N(C)CC3)=O)COC2)ccc(Cl)c([N+](=O)[O-])c1 99588,C1(NC(c2cc(C)oc2)=O)CCCCN(C(C2CC(OC(C)(C)C)C2)=O)C1 99589,CCC(C)(O)C(=O)N(CCCNC(C1C(C(F)F)C1(C)C)=O)CCO 99590,CC(C)CCCC(C)C(=O)NC1CC(C(F)C(=O)NCCc2c[nH]nc2O)C1 99591,N1(C(c2cc(Cl)c(Cl)cc2O)=O)CCCC2(CCC2O)C1 99592,c1(-n2c(C(c3n(CC)ccn3)NCCn3cncn3)nnn2)ccc(Cl)cc1F 99593,Cc1ncc(Br)c(N2CCOC(C(=O)NC(c3ccc(F)cc3)CO)C2)n1 99594,c1(CCCC(=O)OCC(CSCC)O)ccc(Oc2cc(F)cc(Br)c2)c(F)c1 99595,Cc1csc(Cl)c1C(=O)NCC1CCN1C(=O)CC1COCCN1CC(F)(F)F 99596,N1(C(C2(C)CN(C(CC(CC)O)=O)C2)=O)CCOC(C)CC1 99597,c1(COC)cncc(C(=O)N(C(C)CN(C(=O)CCc2cccs2)C)C)c1 99598,c1(CC)cc(C(=O)NCC(C)(C2CC2)NC(c2cc(C)[nH]n2)=O)ccc1O 99599,CC1SCCCC1C(N1CCC2CC12C(=O)NCCNC(=O)CO)=O 99600,Cc1cn2ccc(C(N3CCC(Cc4cn(CCO)nn4)C3)=O)cc2n1 99601,N1(C(C2C(C)(C)C2)=O)CCN(C(c2ccnc(C3CC3)c2)=O)C(c2cccs2)C1 99602,Cc1nc(Cl)ncc1NC(C1CCCN(C(C2CC(C)(C)C2)=O)CC1)=O 99603,N1(C(C(C)S(N)(=O)=O)=O)CC(NC(=O)C(F)(F)C2CC2)CC12CCCCCC2 99604,C(c1ccccn1)=C(C)C(=O)NC1CCC(C)(CNC(c2ccncc2)=O)C1 99605,c1(C(=O)NCCC2CC(NC(C(C)O)=O)C2)sccc1C(C)(C)C 99606,CC1CCN(C(c2ncsc2C2CC2)=O)CC1NC(=O)CSc1cn[nH]c1 99607,C(CC(C(C)C)NC(c1nnnn1C1CCOCC1)c1cncs1)OC 99608,C=C(C)CC(C(=O)NCC1(C)CNC(=O)O1)NC(=O)Cc1cnnn1C 99609,N1(C(C)=O)CC(C(=O)NC2CC2C(=O)NCCN(C)C2CC2)(CO)C1 99610,C1(CCNC(c2cnn(C)c2Cl)=O)CCN(C(=O)Cc2cc[nH]c2)CCC1(F)F 99611,c1(C(N2CCC(CC)C2C(=O)NCCc2ccncc2)=O)cnc(O)cc1C 99612,C1(NC(C=CCN(C(=O)CCOC2CCCC2)C)=O)CCC(F)(F)C1 99613,C1(CNC(C(COC)N(C)C)=O)CCCC2(CN(C(=O)C(CC(C)C)OC)C2)O1 99614,S(=O)(=O)(c1c[nH]ccc1=NC(Cc1cccs1)CO)NCCC(CC)C 99615,C(=O)(C1c2c[nH]nc2CN1C(C1CCC1C)=O)N1CCCC(C)(OC)C1 99616,N1(C(C(C)n2cccn2)=O)CC2CCC(C1)N(C(=O)CCc1cc(F)ccn1)C2 99617,N1(C(C(C)CF)=O)Cc2ccccc2CC1CNC(=O)C(c1ccccn1)O 99618,N1(C(C(CCOC)NC(=O)C=Cc2ccsc2)=O)CCC2(CCC(O)C2)C1 99619,c1(OC)cc(C(=O)NCCN(C(=O)COCCOCCO)C)[nH]n1 99620,C1(C(=O)NCC2(F)CC(NC(c3cnc(Cl)s3)=O)C2)CC2C=CCC(C1)C2 99621,O=C1NC(=O)C(CNC(C2CC23CC(NC(c2[nH]ccc2C2CC2)=O)C3)=O)N1 99622,C1(NC(c2cccnc2N2CCCCC2)C)CCN(C(=O)C(C)(C)CO)CC1C 99623,CCC1=NOC(C(=O)N(C2(C(=O)NC3CCNC(=O)C3)CCC2)C2CC2)C1 99624,C(CC(C(C)(C)C)NC(C1(OC(C)C)CCC1)=O)N(C(C(C)=C1CCC1)=O)C 99625,N1(C(C2(CC)CCOCC2)=O)C2CCC1C(NC(=O)C(C)Sc1ccccn1)C2 99626,C(=O)(CC(COC)NC(C1CCC(C)O1)=O)NC(C12CCC(CO1)C2)C 99627,C1(N(C(CC2(CCN)CC2)=O)C)CCN(C(c2cncnc2)=O)CC1.CSC 99628,C(=O)(CCC(C(C)O)NCc1ccc(N(C)C)cc1F)OC 99629,N1(C(c2c(C)cc(C)[nH]2)=O)CC23CCCC2(C1)CN(C(=O)C=C1CCSCC1)C3 99630,CC1CN(C(C2CC(C)(F)C2)=O)CCCN1C(c1cnc(C(F)(F)F)nc1)=O 99631,Cc1ccc(S(=O)(=O)Nc2cccc3nncn23)cc1NC(c1ccco1)=O 99632,N1(C(CN(C(C(C)C)=O)C)=O)CCC(CNC(=O)C(C(C)C)N(C)C)C12CC2 99633,C(=O)(CCCC(C)(C)C)N1CC(CC)N(C(=O)C(C)NC=O)CC1 99634,C1(CCCNC(c2cccn2Cc2cccs2)=O)CCCN1C(=O)CC1CCC1 99635,c1(C(=O)NC(CC)CNC(c2nc(=N)cc[nH]2)=O)ccc(NC)c(F)c1 99636,Cc1nc(Cl)nc(N2CC3CC2(CNC(=O)CC2CCC(C)(C)CO2)C3)c1[N+](=O)[O-] 99637,Cc1c(C(=O)NC2COCC2NC(=O)Cn2cnccc2=O)[nH]c2c1CCCC2 99638,c1(CCC)nc(C2CC2)ncc1C(=O)NCCN(C(=O)C(F)(F)CC)C 99639,C(C)(CC(C)(C)C)(c1nnnn1C(C)(C)C)NCc1nccc(C)c1 99640,c1(C(=O)NCC(CNC(=O)CCc2ncc[nH]2)F)ccc(C2SCCS2)cc1 99641,c1(C(C)=O)c(NC(=O)C=Cc2c(Cl)cccc2Cl)c(C#N)c2n1CCCC2 99642,CC(C)C(C)(Cc1ccccc1)C(=O)NCCc1ccccc1O 99643,c1(CC)cnc(C(=O)NC(c2cccc(C)c2)CNC(=O)C(=O)C(C)C)nc1 99644,n1(CC)nc(C(=O)NC2CCC2NC(=O)C(C)CC(F)F)c2c1CCOC2 99645,Cc1cc(NC(C2CC2C(=O)Nc2nc(Br)ccc2O)=O)ccc1Br