SMILES CC1(C(N2CCC2Cn2cc(C3CCCOC3)nn2)=O)CCCC1(F)F N#CC1(C(N2CCCC(N3CCN(C(C4(O)CCCC4)=O)CC3)C2)=O)CCOC1 C1(C)(CNC(C(C)COCc2ccccc2)=O)CN(C(=O)CC(=O)NC)CCO1 N1(C(C2C=CCN(C(CCC(C)(C)C)=O)C2)=O)CCC2(CNC(=O)N2)C1 C1(C(=O)Nc2nc(C)sc2)CCC2(CN(C(c3nnc(C4CC4)o3)=O)C2)O1 c1(C(N2C(CNC(C(CSC)O)=O)C=CC2)=O)cn(C2CC2)c(C)cc1=O Cc1cc(NC(=O)C=CC(C)NC(c2c(C)cccc2O)=O)cc(Cl)c1 c1(OC)c(F)ccc(C(N2CC(c3ccc(Br)cc3)CC2C)=O)c1F N1(C(C2N(CC#C)CCC2)=O)CCC(NC(c2c(C)cccc2Cl)=O)CC1C CCCC(C(=O)NCCC1CCC2CC12)NC(C1C=CCC1)=O C(=O)(C(C(C)C)NC(=O)CCCc1cnn[nH]1)NCC=C C1(NC(c2c(C)[nH]cc2)=O)CCCN(C(=O)C(C(C)C)NC=O)C1 N1(C(C(CCCOC)NC(c2c(C)cc(CC)o2)=O)=O)CC2(CCCCCC2)C1 C1(C(=O)NCCc2ncccn2)CCCN(C(c2cccc(C(F)(F)F)c2)=O)C1 N1(C(C(C=C)(C)CC)=O)C2COCC1CC(NC(C1CCOC1)=O)C2 C(=O)(C1=CCCO1)N1C(C(C)(C)CNC(=O)CSc2cn[nH]c2)CCC1 c1(C(=O)NC(CC)CNC(c2cnn3c2OCC3)=O)cc(F)c(C)cc1Cl C1(CC)(NCC(c2csc(=N)[nH]2)=O)CCCC1 CC(CCc1ccco1)N=c1[nH]c(=N)[nH]c(=NC(CCO)C2CCC2)[nH]1 c1(N2CC(CC(C)NC(C3C(OC)CCC3)=O)C2)ncc([N+](=O)[O-])cc1CO CON(C)CCNC(=O)C(C1CCC1)NC(=O)CN(CC(C)(C)C)C C#CCC(C)C(=O)N1CCC(C)(NC(c2ncn(C(C)(C)C)n2)=O)C1 c1(C(=O)NCCN(C)C(C2CCCCC2C(C)(C)C)=O)ccncc1Br N1(C(C(COC)C)=O)CCN(C(c2ccnnc2S)=O)CC1CF c1(C(N2CC(CCCNC(CCC(C)SC)=O)OCC2)=O)cc(O)ccc1Cl c1(C(=O)OC)c(=NC(=O)COCCOCCOCCOCCO)[nH]n2cccnc12 c1(C(N2CCC(O)(CCNC(c3cn(C)c(O)n3)=O)C2)=O)cc(Cl)c(F)c(Cl)c1 C12(CCCOC1)C(=O)NC2.c1(CN(C)C)cncc(-c2ccoc2)c1 C1(CNC(CC(CC)C2CCC2)=O)CC2CCC1N(C(C1CC1C#N)=O)C2 c1(C(=O)NC2CC(CNC(C(COC)N(C)C)=O)C2)ccc(C)cc1SC N1(C(C2(CC#C)CC2)=O)CC(C2CC2C(=O)Nc2ccccc2C(C)C)C1 C(=O)(CCCCC(F)(F)F)N(C)CC1CN(C(=O)CSCC2CCCO2)CCO1 C1(CNC(C(CC)(C)C)=O)CN(C(C2CN(CC(F)(F)F)C2)=O)CC1(F)F C1(CNC(C(CCC)OC)=O)CC2CCCC2N1C(=O)COCCCF N1(C(CCNC(=O)OC)=O)CC(NC(c2cc(C(F)F)nn2C)=O)C(C)C1 N1(C(C2N(S(CC)(=O)=O)CCC2)=O)CCC(C)(CCNC(=O)Cc2nc[nH]n2)C1 N1(C(C2(C(=O)OC)CC2)=O)CCCC(C)(NC(=O)CCC2(C)CCC(=O)N2)C1 c1(NC)cc(C(=O)N(C2CCC(NC(C3CN(C)C(=O)N3)=O)CC2)C)cc(Cl)n1 c1(C(N2CCCN(C(C3CCC(C)S3)=O)CC2)=O)coc2c1C(=O)NCCC2 c1(C(=O)NCC2C(NC(C(C(=C)Cl)(C)C)=O)CCC2)cnc2c(cnn2C)c1N c1(CC)oc(C(=O)NC2CCC(F)(CNC(C3(O)CCOCC3)=O)C2)cc1C N1(C(CCC(C)(F)F)=O)CC(C)(C)CCC1CNC(c1ccc(C2CC2)o1)=O c1(C(N2CCC(NC(c3cnc(SC)n3C)=O)C2C)=O)ccc2c(c1)COC2 c1(NC(C)CC(F)(F)F)ccc(N=c2c(I)c[nH]c3ccccc23)cc1 N1(C(C(C)(C)CF)=O)CCC(C2CCN(C(c3ccco3)=O)CC2)C1 CCCCC(C)(F)C(=O)NC1CCN(CCNC(=O)C(F)=CCCF)CC1 c1(NC(N2C(CC)C(C(=O)O)CC2)=O)cnc(Cl)c(F)c1 N1(C(CN(CC(C)C)C(C2CCC(C)C2)=O)=O)CCC(CC2CC2)CC1 N1(C(C2(C#C)CC2)=O)C2CCC1C(C)C(NC(=O)Cn1ncnn1)C2 CC(CC(=O)N1CCN(C(C2(C)COC(=O)OC2)=O)CC1CO)C(F)F C1(C(=O)NCCCC(C)NC(C2COCCN2C)=O)Cc2ccncc2N1 C#Cc1cccc(CCCNC(C(=O)O)C(C)C)c1 Cc1cc(C(=O)NC2CCCC2NC(=O)C(C)(C)n2cc(Cl)cn2)cn(C)c1=O C(CS(=O)(=O)CC(=O)N1CC(NC(=O)CSc2cnn(C)c2)CC1C)OC CCCCC(C(=O)N(CCCO)CCC)NC(c1ccc(C(N)=O)[nH]1)=O N1(C(CC(CC)SC)=O)C2CCCC1CN(C(=O)Cc1cccc(OC)c1Cl)C2 C(C(=O)N1CCN(CCNC(c2ccccc2O)=O)CC1)(C(F)(F)F)OC(C)=O C(=O)(CCCC(=O)N(C)C)N1CC(NC(c2c(NCC#C)nccc2)=O)C(C)C1 N1(C(CC(=O)NCC#C)=O)CCC(C)C(N(C(=O)C(=O)NCC)C)C1 C(CCCCC(=O)NCCC1(O)CN(C(C2CC2CNC2CC2)=O)C1)N(C)C CC1CC(CNC(=O)Cn2cnnc2)CN1C(C1CC(F)(F)CS1)=O N1(C(=O)CSc2ccccn2)CC2=C(C1)CN(C(C1CCCN1CC1CC1)=O)C2 N1(C(C2(CC#N)COC2)=O)CCCC1CNCC1(C2CCCO2)CC1 Cc1cc(C2CCC2)ccc1C(=O)NCC1(O)CN(C(=O)C(C(C)C)N(C)C)C1 C1(CC(F)(F)F)(NCC2(C3CCCO3)CCC2)CCCC1 C1(C)(COC)CC(NC(c2ccn(C)c2)=O)CN1C(=O)CC1(C)CCOCC1 N1(C(COC2(C)CN(C(=O)CS(N)(=O)=O)C2)=O)CCN2CCOCC2C1 C1(C(=O)Nc2c(C(=O)OCC)n[nH]c2)CC(F)CN(Cc2csc(Br)n2)C1 CCC(C)(C#N)C(=O)N1CCC(O)(CCNC(c2nnn(C)c2C(F)F)=O)CC1 C1(NC(C(CC)CC)=O)CCCN(C(=O)Cn2ccccc2=O)C1CC C(=O)(CCS(C)=O)NC(CC)CNC(c1ccc(OC)s1)=O C1(F)(C(=O)NCC(CC)n2cccn2)CCCN(C(=O)C(CC2CCC2)OC)C1 Cc1cccc(NC(=O)CC2CCN(C(=O)C(O)C(C)C)CC2)c1O C1(F)(CNC(=O)CCC2CC2(F)F)CCC(NC(c2cccnc2O)=O)C1 Cc1nn(C)c(F)c1C(N1CC(NC(c2scnc2C(C)(C)C)=O)CC(O)C1)=O N1(C(c2nccc(C)n2)=O)CC2CC(NC(=O)C=CC3CCCO3)C2C1 C(C(N=[N+]=[N-])C(=O)NCC(O)CNC(c1cnc(C2CC2)s1)=O)OCC C(CC(C(=O)NCc1ccc(C)cn1)NC(=O)Cc1cnc(C)n1C)=CC c1(C(C(=O)NC(C)C)N(C(C)C(C)C)CC)ccc(Br)c(F)c1 C1(CNC(c2cc(CNC(C3(CC)CCOC3)=O)sc2)=O)CCCCN1C c1(Cn2cc(C3N(C(CS(N)(=O)=O)=O)CC3)nn2)nc(O)c2sccc2n1 C#CC1CCN(C(C2C(NC(C3(SC)CC3)=O)C2(C)C)=O)C1 N1(C(C(CC#C)NC(c2oc(C)cc2C)=O)=O)CCC2(CCCOC2)C1 CCCC(C(=O)NCC12CC1CN(C(c1cc(C)ccc1N)=O)C2)S(N)(=O)=O Cc1cc(CC(=O)NCC2CN(C(C3C=CCC3)=O)CCO2)n(C)n1 C1(CNC(C(F)=CCC)=O)CN(C(C)=O)CC12CCOCC2 c1(OCC(=O)N(C)Cc2cn(CC=C)nn2)ccc(C(C)CC)cc1 N1(C(c2c(CC)nc(C)s2)=O)CC2CCC1C2NC(=O)CSCC(=O)OC Nc1cc(Cl)c(Cl)cc1C(=O)NC12CC(C1)N(C(=O)CSc1n[nH]c(O)n1)C2 N1(C(C2(OC)CCCSC2)=O)CCC(C2(NC(=O)C(C)C3CCC3)CCC2)CC1 c1(-c2ccc(C(C)OCCOC)o2)nc(C(C)O)nn1CC(C)(C)CO c1(C(=O)NCC2CC(NC(C(n3ccc(C)n3)C)=O)C2)cc(F)c(C#N)c(F)c1 CC(C)(CCCCNC(=O)C(CC(F)(F)F)C(C)(C)C)C(=O)NNC(=O)C1CC1 c1(-c2cccc(C)c2)nc(=NC2CC(NC(C3C=CCCC3)=O)C2)s[nH]1 C1(C)(CNC(c2c(CC)occ2)=O)CC(F)(F)CN1C(=O)COCC1CCCC1 C1S(=O)(=O)CC2CS(=O)(=O)C(=O)N(CCOCC)ON=C1N=C2CCC(=O)OC O=C1NC(=O)C2(CC(C(=O)NC3(CCNC(=O)C4=CCCS4)CCC3)C2)N1 c1(OCC=CC(=O)NCCN(C(=O)OC(C)(C)C)CC)ccc(C=O)cc1 Cc1cc(Cl)cc([N+](=O)[O-])c1C(=O)NC1CC(O)CN(C(=O)C2=COCCO2)C1 N1(C(CCCOCC)=O)CC(C)N(C(c2cc(C)n(C3CCC3)n2)=O)CC1C Cc1c(Cl)cc(C(=O)Nc2ncc(CCNC(c3ccc(I)c(F)c3)=O)s2)cc1Cl N1(C(C(COC)NC(C)=O)=O)CCN(C(=O)C(C)N(CC(F)(F)F)C)CC1 C1(C)(CNC(C2(C(C)C)CC2)=O)CCCN(C(C2NC(=O)OC2C)=O)C1 C(CCC1CC1)(C(=O)NOCC(O)C(C)C)NC(C(CC=CCC)C)=O C1(C(=O)NC(C)C(N)c2ccco2)CCn2ccnc2C1 c1(CCN(C(CN(C(=O)NCC(C(F)(F)F)OC)C)=O)C)ccc(F)cc1F N1(C(C(CCCC)C)=O)CC2COCC2(C(=O)N(CC(O)COCC)C)C1 N#Cc1ccc(C(=O)NC2CC23CC(NC(c2ccoc2Cl)=O)C3)c(F)c1 c1(NC(C)=O)ccc(CC(=O)N(C2CN(C(=O)COC(F)F)C2)C)cc1 C(=O)(C1CCc2nccn21)N(CCCC(=O)N1CCC(CSC)C1)CC c1(OC)ccc(C(N2CCCC(O)(CNC(=O)CN(C)C3CC3)C2)=O)cc1C Cc1ccc(Br)c(C(N2CCOC(C(=O)Nc3cscn3)C2)=O)c1F Cc1cc(-c2ocnc2C(=O)NCC2CCC2NC(=O)CCC2CCCC2)on1 CN1CCc2cc(C(=O)NC(CNC(=O)CCn3cnnn3)CO)sc2C1 C1(C(=O)NCC(CC)n2cccn2)(OC)CCN(C(=O)CN2CC=CC2)C1 C1(C(=O)NCCCCCNC(C(C(C)O)N(C)C)=O)C2CC3CC(C2)CC1C3 C12(CNC(c3cccnc3CO)=O)CC(CO1)N(C(C1CCCS(=O)(=O)C1)=O)C2 C1(CCNC(CC(CC2CC2)NC(CC2C(CC)C2)=O)=O)CCCC2(CCC2)C1.C C1(NC(CC2CC(OC)C2)=O)CCCN(C(c2ccc(C(F)(F)F)[nH]2)=O)C1C C1(C(N(CCNS(C)(=O)=O)CC2CC2)=O)CCn2ccnc2C1 N1(C(Cn2ccc(C)c2)=O)CCCC2(C)CCCCC12 C1(C(=O)NC2(CO)CN(C(=O)Cc3ccccc3Cl)C2)(COC)CCC(=O)N1 C1(NC(C2(COC)CCC2)=O)CC2CC(NC(=O)CN(S(C)(=O)=O)C)C1C2 C(=O)(C#CC1CCOCC1)N1CC(NC(COc2cccc(C)c2C)=O)C(C)C1 c1(NC(c2c(C)cccc2)C)ncccc1S(=O)(=O)NCCCn1cnnn1 N1(C(C=CS(C)(=O)=O)=O)CC2CCC(N=c3cc(Cl)nc(C4CC4)[nH]3)CC2C1 C1(CN(C(C)(C)C(=O)NC2CC2)C)CSCCN1C(C1CCOC1C(F)(F)F)=O C(C(C)C)(C(C(=O)NCCCF)N1CCCC(C)(C(F)(F)F)C1)OC N#Cc1cn(C2CC2NC(N)=O)c(=O)n(C(=O)c2ccccc2Cl)c1=O CCC(CNC(=O)Cc1c[nH]nc1C)(CC)C(=O)N(CCS(N)(=O)=O)C Cc1nn(C)c(C)c1NC(C1CCC(CNC(C2(CC(C)C)CC2)=O)C1)=O c1(OCC(=C)C)cc(CNCc2snnc2C(C)C)ccc1C(F)F CC1CN(C(=O)CC2CCOC2)CC1CNC(c1c[nH]nc1C1CCOCC1)=O C1(NC(c2ccnc(OC)n2)=O)CCN(C(c2c(Cl)csc2Cl)=O)CC1O N1(C(c2cc(OC)cc(Br)c2)=O)CC(NC(C2C3COCC23)=O)C2(CCC2)C1 C=CCC(C)(C)CC(=O)N1CC2CC(NC(=O)CC3CCCNC(=O)C3)C2C1 C1(NC(CCCc2onc(C(C)C)n2)=O)CC2C1CCN2C(=O)CC(C)C(C)C c1(C(=O)NCC2N(C(C=COCC)=O)CCC2)c(C)cc(O)cc1C N1(C(C2(NC(C)=O)CCC2)=O)CCC2CC2(C(=O)NC2CN(C)CC2(C)C)CC1 C1(C(=O)NCCC(C(C)C)NC(=O)CSCC(F)(F)F)CC2CCCCCCC12 N1(C(CCCC)=O)CC2CC(C)N(C(C3CCNC4(CCC4)C3)=O)C2C1 C1(CC)CCN(C(=O)C(COC(C)(C)C)N(C)C)C1CNC(C1CCOCC1)=O c1(CC(N2CCC(C#N)(c3cc(F)cc(F)c3)CC2)=O)csc2ccc(Cl)cc12 CC1(C=CC(=O)NCC2CN(C(=O)C(F)C(F)(F)F)CC2(F)F)CCOCC1 C(=O)(C1=CCC(F)(F)CC1)NC12CC(CNC(C3(OC)CCSC3)=O)(OC1)C2 c1(CC(N2CC3C(CN(C(=O)CO)C)C3C2)=O)c(F)cc(Br)cc1F C1(NC(c2cc(Br)cnc2S)=O)CN(C(c2ccsn2)=O)CC12CC2 C(Cn1cncn1)(C(=O)N=c1cc2n([nH]1)CCCC2)NC(C1CCC(=O)C1)=O C1(OC)(CNCC(=O)Nc2ccc(=O)n(CC(F)(F)F)c2)CC(C)CC(C)C1 c1(C(=O)NCC(CC)(CC)NC(C(CCC)OC)=O)nc(N)cc2ccccc12 C1(C(=O)NCC(CNC(c2ccc(C)n2C)=O)O)CC=C(C(C)C)CC1 c1(CNC(c2ccc(C(C)=O)[nH]2)=O)ncc(C(=O)NC2CCC2C)cn1 C1(NC(CCCCC)c2nnnn2C2CCOCC2)CCc2nncn2C1 C1(N(CCCNC(=O)Cn2cc(-c3cncs3)nn2)C)CCC(F)(F)CC1 N1(C(C(CC)(C)O)=O)CCN(C(=O)Cc2nc(-c3ccsc3)no2)C(C(C)C)C1 Cc1cc(C(=O)NC2CCCC(CNC(c3ocnc3C(C)C)=O)C2)nn1C C1(C(=O)NC(c2nc(=O)o[nH]2)C)COCCC1NC(=O)CC1C=NN(C)C1=O c1(CC(=O)N(CC(C)O)CCNC(C2(F)CC2C)=O)nccn1C C1(CC(=O)N(CC#C)CC)CN(C(=O)C(C)N(C)C(C)=O)CCC1C Cc1cc(N2CCC(C3(NC(c4cnc(O)nc4O)=O)CC3)C2)nc(C)c1C#N C#Cc1cn(C)nc1C(N1C2CCC1C(NC(=O)CCn1cc(C)cn1)C2)=O c1(C(N(CCN(C(CC(C(C)C)OCC)=O)C)C)=O)cc(Cl)c(F)cc1O CCCCC(C(=O)N1CC(C(=O)OC(C)(C)C)CC1C)SC N1(C(C(CC)OC2CCCC2)=O)CC2CC2(CNC(c2cccnc2S)=O)C1 C1(C(=O)NC2CCCC2CCOCC)(CC)CCCN1C(=O)CN(C)C(C)C C(=O)(C(C)CC(F)(F)F)NC1CC(C(=O)NC2(C(N(OC)C)=O)CC2)C12CCC2 c1(C(=O)NCCN(C(=O)C(O)Cc2cc(Cl)cc(Cl)c2)C)coc(S(C)(=O)=O)c1 C(=O)(CCCCC(F)(F)F)N1CC(C2CN(C(C3(CC#C)CCCCO3)=O)C2)C1 Cc1cnn(C)c1CC(=O)NC1CCCC1NC(=O)CCOCc1ccccc1 c1(C(N2CCC(C)(CC(=O)NCCN3CCC3)C2)=O)ccc([N+](=O)[O-])o1 c1(C(N(C2CCN(C(c3csc(C)c3)=O)CC2)CC#C)=O)cncc(F)c1 Cc1cc(C(=O)NC2C3CN(C(=O)CC4COC(C)(C)CO4)CC23)c(C)nc1C N1(C(CN(C)CC)=O)CC2CCCC(NC(c3cccnc3Cl)=O)C2C1 CCCC(C(F)(F)F)NC(C1(CC)CCN(C(C23COCC2C3)=O)C1)=O C1(CNC(C(C)Cc2ccco2)=O)CCC(N(C(=O)CCSC(F)(F)F)C)CC1 c1(C(=O)NC2C(C(NOCCOC)=O)COCC2)ccnc2cc[nH]c12 C1(C(N(C(c2ccc(OC)cc2)C(=O)O)C)=O)Cc2cc(C)ccc2S1 c1(C(N(C(CCNC(C2(CC)CCCC2)=O)C)C)=O)cnc2cc(C)ccn12 c1(C(=O)NCC2(O)CN(C(C(C)NC(COC)=O)=O)C2)csc2c1CCC(C)C2 c1(NC(C2CC(F)CN2C(c2c(O)cccc2F)=O)=O)ccn2ncnc2c1 CCC(CC)C(CNC(N1CCC(CC(N)=O)(CO)CC1)=O)N(C)C O=C(CCC(F)(F)F)NCC=CCNC(C1CCCS1(=O)=O)=O C1(CNC(CCC(C)(C)OC)=O)CCN(C(=O)CCC(C)(C)C#N)CCC1(F)F C(C1=NOC2CCCC12)NC(C1N(C(c2c(C)c[nH]c2)=O)CCC1)=O CC(C1CCCCC1)=CC(=O)N(CC(O)CN(C(=O)CN1C(=O)CNC1=O)C)C Cc1cc(=O)c(C(=O)NCCCCN(C)C(c2cn3cccnc3n2)=O)cn1C N1(C(c2ccc(OC(C)C)cc2)=O)CCC2(NC(c3cc(F)n[nH]3)=O)CCCC12 C1(C)(CNC(C=C(COC)C)=O)COCCN(C(=O)CC(=O)NC2CC2)C1 CN1Cc2cc(NS(=O)(=O)c3ccc(N4C5C=CCC4CC5)nc3)ccc2C1=O C1(NC(CCCC=C)=O)CCN(C(C2(CSC)CC2)=O)CC(C)(C)C1 N1(C(Cc2c(C)nsc2)=O)CC2CN(C(=O)CNC(=O)Cn3cncn3)CCC12 N1(C(CC=C)=O)CCC(CC=CC)C1C(=O)NCCN1CCCC(O)C1 CCC(C)CC(C)N(c1cc(NCCCCn2nc(C)cc2C)ncn1)C C1(NC(CSC(C)C)=O)CCCC(NC(C2COCCOC2)=O)C1 C1(=CC(=O)NC2CC(NC(C3C(C)(C)C3)=O)C2)CN2CCC1CC2 CC1(C)CC(NC(=O)CCc2ncc[nH]2)CCN(C(C2(C)CCOC2)=O)C1 c1(OC)ccnc(CNC(C2CC3CCCC23)=O)c1OC CCC(CC(=O)NC1(CCOC)CCN(C(c2snc(O)c2Cl)=O)C1)C(F)F C(=O)(C(C(C)C)n1ccc(C)c1)NC(C1(OCC)CCC1)c1nn[nH]n1 c1(C(C(=O)NC(CC)C)N(C2CCC(F)(F)C2)C)ccc(F)c(I)c1 C(=O)(C(C)(CO)OC)NC(CNC(c1cn(CCC)nc1)=O)C1CCC1 CC(C)(C)C(C#N)C(=O)NC1CC(O)C1CC(=O)NCCCO C1(C(=O)Nc2ccc(SC)c(F)c2)COC2(CCN(C(C3(Br)CCC3)=O)CC2)C1 c1(CC(=O)NC2CC(C)N(C(c3c[nH]c(=O)cn3)=O)CC2)ccc(F)c(F)c1F C(=O)(C1=Cc2ccccc2C1)N1CCC(C)C(NC(=O)Cc2nnc(O)s2)C1C N1(C(CCNC(=O)NC)=O)CCCC2C(CCCN2C(c2ccoc2)=O)C1 CC1=C(C(=O)N2CCCCC2C(=O)NC2CC3C(C2)C3(F)F)CCCO1 c1(OC)cc(C(N2CC(F)(F)C2c2ccccc2)=O)ncc1-c1cnoc1 CC(C)(O)CCCC(=O)N1CC(CNC(c2cncc(O)c2)=O)C1 c1(C(N2CCC(NC(C3N(CC)CC3)=O)C2)=O)cccc(NC(=O)OC)c1 N1(C(Cn2ccc(C)n2)=O)CCN(CC(C)NC(=O)C(C)(C)CC2CCC2)CC1 C1(CC(=O)NCC2(NC(=O)C=Cc3ccccc3)CCOC2)CCCOCC1 N1(C(C2C(C(=O)OC)C2)=O)CCCCC1CN(C(=O)CC1CC2(CCC2)C1)C CC(C)C(O)CC(=O)NC(CC1CC1)C(=O)NCCSCCCO C12(C(=O)NCC(C3(O)CN(C(c4cc(C)n(C)c4)=O)C3)(C)C)CCCC1C2(F)F c1(CC)ccc(C=CC(=O)NCC2(OC)CN(C(C3CC3Cl)=O)C2)cc1 C(C)(CC(C)NC(=O)CC(C)O)NC(C1CN(CC(C)C)C1)=O N(C1CCc2cc(CNC(=O)C(=O)Nc3ncc[nH]3)ccc21)C(CCC(C)C)=O c1(C(=O)NC(c2cncc(C(F)(F)F)c2)C)coc(S(C)(=O)=O)c1 c1(C(=O)NCC2(COC)N(C(C(CC)n3cccn3)=O)CCC2)cccc(F)c1 N1(CC(=O)NCCCN(CCO)C(c2ccsc2)=O)CCSCC1 Cc1cc(O)cc(=O)n1CCC(N1CCC(C)C(NC(C2CC3CC2C3)=O)C1)=O C1(CC(=O)N(CC(=O)NC)C)CN(C(c2cc(C)[nH]n2)=O)CC1C c1(CC(=O)NCCN(C(=O)CCC=CC(C)C)CC)ccc(OC(C)(C)C)nc1 CCCC(C(O)C(=O)N(C1CC2CC2C1)C)NC(=O)CC(O)CC(C)C c1(CC2(C(=O)NCC3CCN(C(=O)C(O)CC4CC4)C3)CC2)cccc(Cl)c1 c1(C(=O)NCCC2C=CCC2)ccoc1CNC(C1CC1(F)F)=O C1(CCOC)CN(C(=O)C(=O)NC2CCC(C(C)(C)C)CC2)CCO1 C(C(O)CC(F)(F)F)NC(CC1CCC(NC(C2(C)CC2(F)F)=O)CC1)=O C=CCCCCC(=O)NCC(N1CCN(C(C2CC2C2CC2)=O)CC1)=O C#CC1(N(C)C)CN(C(c2cn(CCNC(C3(O)CCSCC3)=O)cn2)=O)C1 c1(C(=O)NC(C2(O)CCN(C(=O)CCc3ccn(C)c3)C2)C)cccc(CO)c1 c1(CNCc2ccc(C)nc2)cc2cccc(Cl)c2s1 N1(C(C(C2CCOCC2)OC)=O)CCC(N(CCO)C(C2CC(F)(F)C2)=O)CC1 C12(C(N3CC(CN(C)C(C4CCCC(=O)O4)=O)OCC3)=O)CCC(CO)(CC1)C2 C(N=c1[nH]c2ccc(Br)cc2s1)C1CC(C)N(C(c2cccc(C3CC3)c2)=O)C1 CC1CCCCC1(CNC(=O)Cn1ccc(O)nc1=O)NC(=O)Cc1cnsc1 c1(C(=O)NC(C2(O)CCN(C(COC(CC)(C)C)=O)C2)C)cc(OC)ccc1F Fc1ccc(CCCc2nc(C3CCC3)nn2-c2ccc(C(F)(F)F)cc2)cc1F c1(COC(C(=O)NCC(CNC(c2cc(CCC)[nH]n2)=O)C)C)ccccc1C C1(CCNC(c2c(CC)cco2)=O)CCN(C(C2CC(N(C)C)C2)=O)C(C)C1 C12(CCNC(c3nc(C)n(C)n3)=O)CCC1CN(C(=O)CSC(C)(C)C)C2 N1(CC2CCN(C)CC2)CC=C(CNC(c2cnn(CCC(F)(F)F)c2)=O)CC1 Cc1c(C(N2CCC3CCC3C2)=O)c2ccccc2n(C)c1=O c1(SC(C)C(=O)NC2(CCNC(C3CC4CC4C3)=O)CCCC2)ccc(Cl)cc1 C1(NC(C(CC)C(C)C)=O)CC2CCCC(C1)N2C(c1nnsc1C)=O N1(C(C2C=C(C)CS2)=O)CCCC(C)(C)C1CNC(=O)CO C1(NC(=O)OC(C)(C)C)CC2CCC1N(C(C1CCC3CCCC3O1)=O)C2 C(CCCCC(=O)NC1CC(NC(C2(C)CCC(N(C)C)CC2)=O)C1)OCC c1(C(N2C(CNC(c3csc(C)c3C)=O)COCC2)=O)nc2c(s1)CN(C)CC2 Cc1nn(C)c(C(N2CCCC(CCNC(=O)CC3COCCO3)C2)=O)c1Cl c1(C(=O)NCCc2ccc(OCCCC)cc2)ccc(F)c(Cl)c1 C(=O)(C(C(C)NC(=O)C(COCC)OC)C(C)C)NC1CN(CCC)C1 Cc1nn(C(C)C)cc1C(=O)NC1CCCC(NC(=O)Cc2ncn(C)c2C)C1 C#CC1(C(=O)NC(CCCCC)C2CC2)CCN(C(=O)CC(CC)SC)C1 N1(C(Cc2n(C)cnc2)=O)CC2(C1)CN(NC1(CCF)CCC1)C2 C1(CC(=O)NCC(CC)C)CN(C(C2CC(=O)CC(=O)N2)=O)CC12CC2 c1(NC2C3(C(=O)OC)CC3CC2)cc(C)ccc1[N+](=O)[O-] C(=O)(C(C(C)C)N1CCC(C)CC1)NCC1(F)CN(C(Cc2nnc(C)o2)=O)C1 c1(N2CC(C)(CCO)OCC2)nc(N2CCOC3(CCCC3)C2)nc2sccc12 c1(C(=O)NC2CC(NC(=O)CC(O)CC3CC3)C2)cnc(O)c2c1NCCC2 N1(C(C(C(C)(C)O)NC(C(c2ccccc2)C)=O)=O)CC2C3C=CC(C3)C2C1 C1(C(N2CC(N(C(C3CCN(C(C)=O)CC3)=O)C)C2)=O)CN2CCC1(C)CC2 CC(C)(CC(F)F)C(=O)N1CCC(O)C(NC(C2CCC=CCCC2)=O)C1 C1(NC(C(C)SC)=O)CCC(CN(C)C(c2conc2-c2ccccc2)=O)CC1 c1(NC(N2C(C=C)COCC2)=O)ccc2cc(C)oc2c1 C1(NC(CCC)=O)CN(C(=O)C(=Cc2ccc(Cl)cc2)C)CC12CCC2 Cn1cc(C=CC(=O)NC2CC2NC(=O)Cc2cc(C3CC3)no2)cn1 Cc1nc(S(C)(=O)=O)sc1C(=O)NC1CCN(C(C2CCC(=O)N2)=O)C1 c1(C(N2CCC(c3c(-c4onc(C)n4)cccc3)CC2)=O)c(F)cc(F)cc1F c1(C(N(CCNC(=O)CCCc2cc(C)no2)CC)=O)n[nH]c2c1CCC2 N1(C(COC(CC)C)=O)CC2(C1)CN(C(=O)CC1CC(COC)C1)CCO2 C12CCCN(CC1)C(=O)N(C)C2.c1(O)ccc(OC)cc1.CCCOC C=C(Br)CC(=O)NCCC1CCCN1C(C1CC1(Cl)Cl)=O C(=O)(C(C(CC)CC)OC)N1CC(C=C)(C(N2CCCC(C)C2CCO)=O)C1 C(=O)(C1=CC2CCCC12)N1CCCC(CCNC(c2c(C)cc(C)o2)=O)CC1 CS(=O)(=O)c1cc([N+](=O)[O-])ccc1NC12CC3CC(C(=O)N1)C2C3 C1(O)(CNC(=O)COCCC2CCCOC2)CCCN(C(=O)CN2CCCC2)C1 N1(C(=O)CCC2CCC2)CCCC12CCCN(C(=O)Cn1ccc(C3CC3)n1)C2 C(=O)(C1CCCc2sccc21)N1CC2CCC(NC(C=C(CC)C)=O)(C1)C2 c1(CN(CC(CC)Oc2ccccc2)CC)csc2ccc(C(=O)O)cc12 CCCCC(CNC(c1nccnc1C(F)(F)F)=O)NC(=O)CN1CCSCC1 N1(C(c2n(C)nnc2)=O)CC(C)(C)C1Cn1cc(CS(C)(=O)=O)nn1 N1(C(C(C2(O)CCCCC2)CC)=O)CCN(C(=O)C(C)CF)C2(CCC2)C1 c1(SCC)ccc(C(=O)NC2CCCC2NC(C2CCOC2C2CC2)=O)cn1 c1(C(N2CCC(CC=C)(C(=O)NC(CO)C3CC3)C2)=O)ccc(=O)n(C)n1 c1(C(N(C2C(C)CCNCC2)C(c2cccnc2)C)=O)cc(S(N)(=O)=O)co1 C(=O)(CC1CCCc2ccccc21)N(C(CNC(C(C)CF)=O)C)C N1(C(CCN(C(=O)CCC2CCCOC2)CCCO)=O)CCOCC2(CC2)C1 C1(C(N2CCC(NC(C(CC)(F)C(=O)OC)=O)CC2)=O)Cc2ccc(F)cc2C1 C(=O)(CCCCCCCCC1CC1)NC1(c2ncc(C)o2)CC1 c1(C(=O)NCC(C)(C)CNC(c2occc2C2CC2)=O)c[nH]c2nc(Cl)ccc12 c1(CC(=O)NC(CNC(C2C(C=C)C2)=O)(C)C2CC2)cc(Cl)c2c(c1)OCCO2 C1(C(=O)NC(c2cccnc2)c2nn[nH]n2)CCc2ccccc2C1 C#CCC(C(=O)NCc1cc(C)ccn1)NC(c1ccon1)=O C1(OC)CC(NC(=O)CCc2ccc(Br)nc2)CN(C(C23CC(F)C2C3)=O)C1 Cc1cc(Cl)c(C(=O)NC(C)CCCNC(c2cc(C(N)=O)[nH]n2)=O)cc1C C=C(C)C(CC(=O)NC1CC1C1CN(C(=O)CSCCCC)C1)OCC C1(C(=O)OCC)CC2CCC(C1C)N2c1cnc(C#N)c(F)c1 c1(C(=O)NCC2(O)CCN(C(C3C(CC)C3)=O)CC2)ccnc2c1CCO2 CCCC(C(O)C(=O)N1CC(CO)C(C)C1)NC(=O)C(F)=C(C)C N1(C(=O)NC(c2ncc(C)s2)CC)CCCC2(CNC(=O)O2)C1 CC(C)CC(O)CC(=O)N(C1CCN(C(=O)CC(F)(F)Cl)CC1C)C Cc1cccc2cc(C(=O)OCC(c3cccc(C(F)(F)F)n3)=O)sc12 N1(C(C(C)CF)=O)CCCC(Cn2cc(CN3CCCC3CO)nn2)C1 C(CCC)(C(=O)N1CC=CC1CNC(C1CC(C(=O)NC)C1)=O)=CCC N1(C(C2C(NC(C(C)C3CC3)=O)COC2)=O)CCC(N=[N+]=[N-])C1 CC(CC(C)NC(=O)C=CC(C)(C)C)NC(=O)CC1(CO)CCC1 C1(CSc2n(C)c(CCCc3ccccc3)nn2)CCN2CCCC2C1 NS(=O)(=O)c1csc(C(N2CC(CNC(=O)Cc3cncnc3)C3CC23)=O)c1 C1(NC(c2ccc(CCC)[nH]2)=O)CCCCC1NC(C1(F)CCOC1)=O C1(NC(C2C(C)(C(C)C)C2)=O)CN(C(c2nnn(C(C)(C)C)n2)=O)CC12CCC2 c1(C(N2CCN(C(=O)CSC3CC3)C3(CC3)C2)=O)ccc2nc(S)oc2c1 Cc1ccc(CCNC(C2(CF)CCN(C(=O)CCc3ccoc3)C2)=O)cn1 CC(CN=c1[nH]c(=NCc2ccc(Cl)nc2OC(F)F)[nH]c2cc[nH]c12)C1CC1 c1(NC(C)=O)cnc(C)c(C(N2CC=CC2CNC(c2ccc(Cl)cc2C)=O)=O)c1 c1(N(C)C)cc(C(=O)NCC2CCC(NC(C3C4CCC3CC4)=O)CC2)ccn1 CCCCC(O)CC(=O)NC(CCOCC)C(N1CCC12CCCCC2)=O n1(CC)nc(C2CC2)cc1C(N1CCC(C)C1CNC(c1nc(C)c(C)[nH]1)=O)=O C1(NC(N2CC(C(=O)NC3C(C)(CC)C3)C2)=O)(CO)CC(C)CC(C)C1 C1(C(=O)NCC2C=CC(NC(C3ON=C(C)C3)=O)C2)CC2CCC1CC2 c1(C(CC)=O)cc(C(N2CCOCC2CCNC(=O)C=CCOC)=O)ccc1F c1(NC(c2cccc(NC(c3c(COC)c[nH]c3)=O)c2)=O)cc(F)ccc1O c1(OC)ccc2[nH]c(C(=O)N(CC(C)N(C)C(c3nc(C)oc3C)=O)C)cc2n1 CCC1=C(C(=O)NCC2CC(CNC(c3oc(CO)nc3C)=O)CO2)CCCO1 C1(NC(c2cc(C)sc2)=O)CN(C(C2CCCN2C(C)C)=O)CC1(C)C N1(C(C2N(C(c3c(C)cco3)=O)CC(F)C2)=O)CCn2ncc(C)c2C1 C1(CNC(C2N(S(C)(=O)=O)CCC2)=O)CC2CCC1N2C(c1ncc(Cl)n1C)=O Cc1cc(C(N2CCC(N(C)C(c3nn(C)cc3N)=O)C2)=O)cnc1C C(=O)(C1=CC2CC=CCC12)N(CC(C)(C)CNC(=O)C(C)(C)CF)C c1(CC(=O)NCC2CC2NC(=O)CCc2cccnc2)cc(Cl)cc(Cl)c1 C1(C)(C(=O)NCC(CC)NC(c2cc(C3CC3)n(C)n2)=O)CCC12CCC2 CCCCCC(O)C(C)C(=O)NCCN(C)C(c1ccc(C(C)C)o1)=O c1(NC(=O)NCCC(CC)C)cnc(C)nc1OC C(=O)(CCCCN(C)C(C1CN(C)CCO1)=O)NCC(C(=O)OC)OC C1(CNC(C2N(C)C(=O)CC2)=O)CC2(CCN(C(=O)CC3CCC(O)C3)CC2)C1 N1(C(C2(NC(CSCCC(C)C)=O)CCSC2)=O)CCC2C(O)CC12 Cc1cc(-c2nc(-c3oc(Br)cc3C)n(CCC(C)C)n2)c(C)o1 C1(CNC(c2c(CC)cc(F)cc2)=O)CC2(CCC2)CN1C(=O)CCCC#N C1(C(=O)NC2(C)CC(NC(=O)CNC(=O)C3CC3)C2)CC1C1CC(F)(F)C1 C(=O)(CCOCCC)N(CC#C)CC1CC1.C1(=O)CCSCCC(C)N1C O=C(NNC(=O)CCOc1ccc(Cl)cc1)C(=O)NC1CCOC1 c1(C(=O)NC2C(C=C)CN(C(=O)C(C)S(C)(=O)=O)C2)nc2cnccc2s1 N1(C(c2cccs2)CNCc2cccc(CNC)n2)CCC2CCCCC2C1 c1(C(c2n(C(CC)C)nnn2)NCCCCOC)ccc(-c2cncnc2)cc1 C(=O)(CCC(O)C(C)(C)C)NCC(CC)NC(=O)CCC(=O)NN(C)C C1(C(=O)NCCCn2cc(-c3cc(Cl)ccc3Cl)nn2)CC2C(C1)C2(F)F N1(CC)C(=O)CCC1C(N1CC(O)(CCNC(C2CC23CCC3)=O)C1)=O CCC(CNC(=O)C(CC(F)F)CC)(CC)C(=O)O c1(C(=O)NCC2(CNC(C3CC(C)(F)C3)=O)CCCCC2)ccc(Cl)cc1F C1(C(=O)NCC(C)N(C)C(c2cc[nH]c(=N)c2)=O)CCCCS1(=O)=O N1(C(CCC2CCN(C(c3cnc(=N)[nH]c3)=O)CC2)=O)CCCC2CCCC12 N1(C(c2c(C)c[nH]c2)=O)CC(C(=O)N(C2CC(F)(F)C2)C)CC(C)(C)C1 N1(C(C(CSC)OC)=O)CCC2CCCC(C1)N2C(c1cc(N)cc(O)c1)=O C1(O)(CNC(C2C(OC)CCCC2)=O)CCN(C(=O)C2=CCCS2)CC1 C(=O)(C1CCc2c[nH]nc21)NC1C(C)N(C(C23CCCCC(F)(C2)C3)=O)CC1 CC1CCN(CC(=O)NCc2cc(C(N3CCCC3c3ncc[nH]3)=O)on2)CC1 CN=c1ccc(C(N2CC=CC2(C)C(=O)NCC(O)COC)=O)c[nH]1 N1(C(=O)NCCN(CCCOC)C)CC2(CCC2O)C1 CC(CC(=O)OC1CCN(C(=O)N(c2ccco2)Cc2cnn(C)c2)C1)C1CC1 Cc1nn(C(F)F)c(C)c1CC(=O)NCC(C1CC1)NC(c1nn(C)cc1Cl)=O C1(CC(=O)N(C2CCCN(C(C3CCN(C)C3)=O)C2)C)COc2ccccc2O1 N1(CCCCC=C)C(=O)CN(CCN2CCCOC(C)C2)C1=O C1(CNC(CC2CCCC(C)O2)=O)CCCCCN1C(=O)CCN1CCCC1 CS(=O)(=O)c1cccc(-n2cc(CONC(c3ccc(Br)cn3)=O)nn2)c1 n1(CC)ncc(C(=O)NC2CCCC2NC(=O)COCP(C)(C)=O)c1C(F)(F)F C(=O)(C(C(C)C)Oc1ccccc1)NC(CC)CNC(c1snnc1C1CC1)=O c1(OC)ccc(NC(=O)C(c2ccnn2C)N(C)Cc2ccsc2)cc1 N1(C(C(C)n2ccnn2)=O)CC(CNC(=O)CCc2cncs2)CC1(C)C C1(C(=O)Nc2ccc(CC)nc2)CCN(C(C2CCC(=O)N2)=O)CC1O C(C)(C)(C#CC(C)(C)O)NC(=O)NC(CC)(C)CO C1(CNC(CCCN(C)C)=O)CN(C(c2cc(C3CCC3)no2)=O)CCC1(F)F CC1CC(NC23CCC(C(=O)N(C)C)(CC2)C3)CC(C)S1(=O)=O C(CC(C(C)C)NC(c1ccc(OCOC)cc1)=O)N(C(C1C(=C)CC1)=O)C C=C(Cl)CC(C(=O)NCC1(C)CCCCO1)NC(=O)CC1OCCC1(C)C c1(C(=O)NCCC2(CNC(=O)C=C(Cl)Cl)CC2)ccnc2[nH]ncc12 N1(C(c2c(CC)n[nH]c2)=O)CCC(C(=O)NC(C)C(F)(F)F)(OC)C1 c1(C(N(CC)CC)=O)cn2c(n1)CN(C(c1ccc(Br)c(C)n1)=O)CC2 N1(C(=O)C(c2ccccc2)O)CCN(C(c2ccnn2C2CCC2)=O)C(CO)C1 Cc1ccc2c(c1)CCC2N=c1ccnc(N(C)Cc2nnc3n2CCOC3)[nH]1 N1(c2ccnc(N(C)CCNc3ccccn3)n2)CCC2(CCSC2)C1 C12(NC(C(=O)N(C)C)=O)CCCC(CN(C(c3cc4c(s3)CCC(C)C4)=O)C1)C2 CCC(CCOC)C(=O)NCC1CCN(c2ncc(I)cn2)C12CC2 C1(NC(C=CC=CC)=O)C2CC(O)C1N(C(=O)CC1CCC3(CCC3)O1)C2 Cc1ccc2c(c1C(=O)Nc1ccccc1CN)CCCN2 C1(CCONC(=O)N(CC(=O)N(CC(C)(C)C)C)CCO)CCC(=O)NC1 N1(C(CC(C)C(F)(F)F)=O)CCC2CCN(C(=O)CCC(=O)c3ccc[nH]3)C2C1 C(C(CC(F)(F)F)NC(=O)Cc1ccoc1)NC(CCC1N(C(C)=O)CCC1)=O CN1CC=C(CC(=O)NCCCCC2CCCN(C(=O)C=CCO)C2)CC1 c1(CC(=O)N(C2CCN(C(=O)CN3CCCC3)C2)CC)cc(C(F)(F)F)nn1C CN1CC(NC(N2CCS(=O)(=O)CC2c2ccccc2)=O)CC(F)(F)C1 C1(CC(=O)NCC(C2CC2)N(C)C(C2CC2[N+](=O)[O-])=O)(OC)CCCC1 OC1CN(Cc2ccc(C3OCCO3)cc2)CCC12CCCNC2 N1(C(c2cc(CNC(C3CCCSC3)=O)ncc2)=O)CC(F)(F)C(F)(F)C1 C1(CC(=O)NCCCNC(c2cc(C(F)(F)F)n[nH]2)=O)CCC2CC12 C(CC1=CCN(C(=O)CCC2CCOC2)CC1)NC(C12CCC(C)(C1)CO2)=O CC(C(C(=O)NCc1nnn(C)n1)N(C1CC(F)(F)C1)C)C1CCOCC1 C1(C(NOCC(CC)C)=O)CCN(C(=O)Cc2ccc(C)nc2)O1 N1(C(C2C(C)(C)C2)=O)CCCC2CN(C(c3cnnn3C3CC3)=O)CCC12 CCC(CC)C(CN=c1nc(N2CCSC(C(C)C)C2)c2c([nH]1)CCC2)OC CC1(C)CC(NC(C23CC(c4ccccc4)C2C3)=O)CCN(C(=O)CNC=O)C1 c1(C(=O)NCC(C)(C)NC(C(CC=CCC)C)=O)ccn2cnc(C)c2c1 C1(C)(C(N2CC(COC)(NC(=O)C(C)N(C)C(C)=O)C2)=O)CC(C)=NO1 N1(C(c2cn(C)nn2)=O)CC(C2CC2)(C(=O)NOCC2CCCC2)C1 N1(C(c2c(C)snc2)=O)CCC(C)(C)C(CNC(C2CC3(CC3)C2)=O)C1 c1(C(=O)NCC(CC(C)C)C)ncc(C(F)F)cc1F CCC(CCOC)C(=O)Nn1cc(-c2ccc(SC)cc2)nn1.C12CC(C1)C2 C(=O)(CC(C)(C)CC(=O)OC)NC1CCC(N(C(c2ccc(CSC)o2)=O)C)C1 c1(-c2nn(CCCS(C)(=O)=O)c(C3CCCCN3C3CC3)n2)cc(F)cc(F)c1 N1(C(c2ccnc(OC)n2)=O)CCC2C(C1)CN2C(c1cc2n(n1)CCCC2)=O c1(C(N2CCC(N(CCO)C(C3CC3C(F)F)=O)C2)=O)ccnnc1O Nc1cc(C(N2CCC(NC(C3C4COCC34)=O)C(CO)CC2)=O)cc(O)c1Cl N1(C(Cn2ccc(C)c2)=O)CCCCC(NC(c2ncoc2C2CCC2)=O)C1 C123C(C4CC1C2C4)NC3.C1(C(=O)OC)CC(C)(NC(=O)CNc2ccccc2)C1 n1(CC)nnc2c(NCC(C3CCCC3)NC(c3ccc(F)nc3)=O)ncnc12 N1(CCC(C)(C)C)CCC2(CC1)CC2NC(c1ccc2c(c1)OCO2)=O C(=O)(C#CC1CCOC1)N1CC(C(C(=O)NCC2CN(C3CC3)C2)OC)C1 c1(C(=O)NCC(CO)NC(c2cnc(SC)s2)=O)ccc(C2CC2)nc1 Cc1cc(Cl)ccc1OC(C)C(=O)NC1CCCN(C(=O)CNC(=N)N)C1 c1(C(N(C2CCN(C(=O)C3=CCC3)CC2)CC#C)=O)cc2ccc(C)n2cn1 c1(C(N(C(CCNC(c2cc(C)c(C)o2)=O)C)C)=O)csc2c1CCCC2 c1(C(N(C)CC2(CNC(C3(CC=C)CC3)=O)CC2)=O)cn2ccnc2cn1 c1(Cc2nc(C)sc2)cccc(C(=O)NC2CC2CNC(=O)CNC(N)=O)c1 c1(C(C(=O)NC(C)CNC(C2CC2Cc2ccccc2)=O)O)ccc(F)c(F)c1 C1(OC)CC(NC(c2cccnn2)=O)C12CCN(C(C1(C)CC(F)(F)C1)=O)CC2 C(=O)(C1=NOC(CNC(C2(C#N)CCC2)=O)C1)Nc1cnc(C(C)C)nc1 C1(CC)CN(C(c2cnn(CCO)c2)=O)CCC1CNC(C1CCC(=O)O1)=O CC1CN(C(=O)Cc2sc(=N)[nH]c2-c2cccs2)CCN1C(C1CCC2CC12)=O c1(C(=O)NCCN(C(=O)C(C)(c2ccccc2)OC)CC)cccc(N(C)C)c1 C12(CCN3CCC1C3)c1nnnn1CCN2.CCCC(C)(C)NC1CCCCC1 c1(C(C)NC(CN2CCOCC2)C(C)C)ccc(C(F)(F)F)cc1 c1(C(=O)NC2C(C(=O)Nc3cc(SC)n[nH]3)C2)cnc(Cl)c(I)c1 Cn1nc(CNC(C2CCCN2C(c2sccc2F)=O)=O)n(C)c1=O N1(C(c2c(C)n(C)cc2)=O)CCC2(C1)CN(C(c1cc3ccsc3s1)=O)C2 C(CN=c1cc(CC2CC2)nc[nH]1)OCCNC(C12OCCC(C)(C1)C2)=O c1(C(N(CCC2CCN(C(CC(CC)C)=O)CC2)C)=O)ccc(Cl)c(N)c1 Cc1c(CC(=O)NC(C)C(=O)NCCC#N)cccc1Br N1(CCNC(CN(C)CC)=O)CCC(NC(c2scc(C)c2Br)=O)CC1 C1(C)(C(=O)NCCCCN(C(C(CC#C)C)=O)C)CCC12CCC2 c1(C(=O)NC2C(CNC(c3cc(C)c(O)nc3)=O)C2)cc2c(C)c(Cl)ccc2[nH]1 N1(C(C(=O)NC(CC)(C)C)C2CC2)CCN(S(C)(=O)=O)C(C)C1 CC1COCCC1C(N1CC(CCNC(c2ccc(C(F)(F)F)o2)=O)C1)=O C(=O)(CCCCC(C)C)NC(c1cn(C)nn1)C(=O)N(CC)CC1(O)CCC1 C1(CC)C(NC(=O)CCc2cnccn2)CCCN1C(=O)CCc1cn(C)nn1 C1(OC)CC2(C1)CN(C(C1(C(=O)NC3CC3C3CCC3)CC(O)C1)=O)C2 N1(C(CCc2ccn(C)c2)=O)CCC2CCN(C(=O)CCC3CC3C(F)F)CC12 c1(C(N(CC(=O)NCC2CCOCC2)CC)C)ccc(F)cc1 C1(CC2OCC(C(N3CCOCC3)=O)C2)COC2(CCC2)C1.c12cc(ncn1)N2 N1(C(CC(C)(C)C)=O)C2CCC1(c1cn(CCOCC3CCCO3)nn1)CC2 N(C(=NCC(C)(C)CC(C)C)N(C)CC1OCc2ccccc21)C(CC)C c1(CC)ccc(C(=O)NCCN(C(=O)Cc2ccsc2C)CCOC)c(C)n1 Cc1ccnc(O)c1C(N1CC(C(C)NC(C2(C)CCN(C(C)=O)C2)=O)C1)=O CC1CC(CC(=O)NCCc2noc(=O)n2C)CN1C(c1cnc[nH]c1=N)=O C1(C(=O)NCCn2cc(C(N(CC(O)CF)C)=O)nn2)CN2CCN1CC2 C#CC(C)(C)C(=O)NCc1cccc(C(=O)NCC2CC2Cl)n1 N1(C(C2C(=O)NCC2)=O)CCCC(c2ccc(F)cc2)C1 C1(C(N(C)CC2(C)CCCC2O)=O)CC(NC(C2C(C)(C)C2(C)C)=O)C(O)C1 C=C=C(C)CC(=O)NCCCN(C(=O)CC1NC(=O)NC1=O)C(C)C CN(C)S(=O)(=O)N1CCC(C(=O)NC2CCCC(c3cccc(Cl)c3)C2)CC1 c1(C(N2CCC(NC(CC(COC)(C)O)=O)C2)=O)cc(Cl)cc(C)c1C CCC(CN(C)C)CC(=O)NCC1(CNC(=O)CSC2CCCO2)CCCC1 Cc1ccc(C=CC(N2CC3CC2(C(=O)NC(C2CCOC2)CO)C3)=O)cc1 C(C(O)C(=O)NCCOCCC(=O)NC(C1CCCO1)CC)=CC O=CN1CCCC1C(=O)NC(c1cccnc1)C(=O)NCCC1CC1 C1(NC(CSCc2nc(C)sc2)=O)CCN(C(C2CCOC2=O)=O)C12CCC2 C1(CNC(C2(CCC)CC2)=O)CN(C(=O)C(C)CN(C)C)CCC12CCC2 Cn1cccc1C(=O)C(=O)NC1CC1NC(=O)CCC1CCOCC1 C1(=CCNC(C=CC=CC)=O)CCN(C(=O)Cc2ccc(CCC)cc2)CC1 c1(C(C)N(C(=O)C(=O)NCC2C=CCCC2)C2CC2)nc(C2CC2)cs1 N1(CC)CCOCC1C(=O)NCCCC(C)NC(c1cc(-c2ccoc2)[nH]n1)=O C1(C(N2C(Cc3cn(CC(C)C)nn3)CCCC2)=O)CCc2nnc(O)n2C1 N1(C(c2n(CC)ncc2)=O)CC2(CC(C(=O)NC(CC)(CC)CCO)CO2)C1 C1(C(=O)NCC2(O)CC(CNC(CCC=CC(C)C)=O)C2)CC2CCC1O2 Cn1cc(CC(=O)NC2CCN(C(=O)CCn3cnnn3)C2)cn1 c1(C(N2CCC(O)(CNC(c3cc4n(n3)CCC4)=O)C2)=O)cncc2c[nH]nc12 c1(CNC(C(C)=C(C)C)=O)nc(C)c(C(N2CCC(F)CC2)=O)o1 c1(C(N2C(CCC(C)(C)NC(C(=O)N(C)C)=O)CCCC2)=O)ncc(Cl)cc1F N1(C(CN2C(C)CCC2)=O)CCC(NC(C2(C)CCCN(C)C2)=O)CC(C)(C)C1 N1(C(c2cc3n(c2)CCCC3)=O)C2CCC1C1CC1(NC(=O)C(F)(F)C(F)F)C2 c1(-c2ccc(C(=O)NCC3(NC(C(CC)N(C)C)=O)CCC3)o2)ccccc1Cl C(=O)(C(O)CNC(=O)CC1(O)CCCC1)NCC(C)(C)N(C)C N1(C(C2C(C=C)C2)=O)CCCC(O)(CNC(c2ccc3ncsc3c2)=O)CC1 C1(NC(CC2(C(=C)F)CCC2)=O)CN(C(c2ccncc2Cl)=O)CCC1O CC1(C(=O)NC2CCN(C(c3cccc(Cl)c3)=O)CC2C(N)=O)CCCCCC1 C1(NC(=O)OC(C)(C)C)CC(S(C)(=O)=NS(=O)(=O)c2cc(C)c(Br)c(C)c2Cl)C1 C=CCCCC(C)(C)C(=O)NCC(C)C(=O)Nc1cnc(C)c(C)c1C O=C1CCCC(C(N2CCN(CC3(NC(C4CCC5(CC5)C4)=O)CC3)CC2)=O)N1 N1(C(CCCCN(C(C)C)C)=O)CC2CCC2(CNC(C2CCCCN2C)=O)C1 c1(C(=O)NCC23CC2CN(C(c2ccco2)=O)C3)cc2c(Cl)cccc2s1 CC1CC(c2nnnn2C2CCOCC2)(NCCc2nc(=O)o[nH]2)CN1C1CC1 N1(C(c2c(C)noc2C)=O)CC(CNC(c2cnc(C3CCC3)o2)=O)C(C)(C)C1 CCC(C)(CC)C(=O)NC(C1CCCC1)CNC(=O)CCCN(C)C CC(C)(C)C#CC(=O)N1CCC(=CCNC(=O)COCC2CCCCO2)CC1 CC1CC(C(=O)NCCCC2CN(C(C3(C#N)CC3)=O)CCO2)=NO1 C1(NC(C(C)(C)O)=O)CCC(NC(C2CCCCC2CC(F)(F)F)=O)CC1 Cc1nccnc1C(N1CCCC1C1CCN(C(=O)C(C2(O)CCCC2)F)C1)=O C1(C(=O)OC)CN(C(=O)Nc2ccc(C(=O)Nc3csc(C)n3)cc2)CCC1O c1(CC(c2ccn(CC)c2)NCc2ncn(C(C)C)n2)ccccc1F c1(C(=O)NC2CCN(C(C(CC)C(C)(F)F)=O)C2C)cc(Cl)cc2ccncc12 N1(C(C(COCC)C)=O)CCN(C(c2c[nH]nc2Br)=O)C2CCCC12 N1(C(c2c(NC(C)=O)cccn2)=O)CC(CNC(C2C(C)C2C)=O)CC(C)(C)C1 c1(C(N2CC(CNC(C(C)C(C)(C)C)=O)C(C)(C)C2)=O)ccc2cc[nH]c2c1F C1(C)(C(=O)NCC(C(C)C)NC(C2CC(C3CC3)C2)=O)CCN(C)CC1 c1(C(N(CC(C)NC(C2CCC(=C)CC2)=O)CC)=O)cn(C)ccc1=O N1(C(C2CSCC(=O)N2)=O)CCN(C(c2ncnc(O)c2F)=O)C(CO)C1 C1(CCNC(CCSCC(C)C)=O)COCCN1C(C1(C2CCCCO2)CC1)=O c1(C(N(CC(C)NC(C2(C)CC2C)=O)CC)=O)cn(C)c2ccc(F)cc12 c12cccc(n1)C(=O)NC2.C1(NC(c2scc(CC)c2)=O)CN(C(C)C)CC1C c1(C(=O)NC2CC(NC(C(COC)CC(C)C)=O)C2)sc(S(C)(=O)=O)nc1C C1(NC(C2(NC(N)=O)CC2)=O)CS(=O)(=O)CC1NC(c1cccc(CF)c1)=O c1(CC(=O)NCC2(C)CCN(C(CCC(CC)C)=O)CC2)cn2ccccc2n1 C1(NC(c2cnc3ccoc3c2)=O)CN(C(=O)C=C2CC2)C2(CCOCC2)C1 c1(C(=O)NCC(CNC(C(C)C2CC2)=O)CO)cccc(-c2ccccc2)c1O N(C(=S)NNC(=S)N(C)c1ccc(Cl)c(F)c1)C(C)C1CC1 C(=O)(C1CCCc2c1ncn2C)NCC1CCN(C(C2CC(SC)C2)=O)C1 C1(c2n(-c3ccc(OC)cc3)nnn2)(NCC2COC2)CC2(CCC2)C1 c1(C(=O)NC(CC)CNC(=O)CC2CCCO2)c(OC)ccc2cccnc12 c1(C2(N(C(=O)C(C)(C)OCC)CC)CC2)ccc(C(=O)OC)cc1 C1(C)(CCNC(C(C2CCC(=O)N2)C)=O)CCCC1.C12CN(C1)C(=O)CO2 N1(C(c2cc(C(C)C)n(C)n2)C(=O)NCCC2CC2)CCN2CCC1CC2 Cc1cccc(C(=O)NC(C)C(=O)NC2CC(NC(C3CC(C)(C)CO3)=O)C2)c1 C1(C(=O)NCCC2(O)CN(C(CCc3nnc(C)n3C)=O)C2)COCC(C)(C)O1 N1(C(C)C)CCOC(C(=O)NC2(CNC(=O)C(C)C(C)O)CCCCC2)C1 C(=O)(C(C)(C)C(=O)NCc1c(-c2cn(C3(C(=O)O)CC3)nn2)cnn1C)N(C)C CN1CCOCC1CC(N1CC(O)(CNC(c2cc(C(C)(C)O)on2)=O)C1)=O c1(-c2cccc(-c3ccc(CN(C4CNC4)C)cn3)n2)c[nH]c2ccccc12 c1(C(C)=O)ccc(C(=O)NCC2(O)CN(C(c3ncoc3C(C)C)=O)C2)cc1C C(=O)(C1CCc2c[nH]nc21)NC1CCN(C(Cc2cn(CC)nn2)=O)C1 c1(NC(c2ccc(NS(C)(=O)=O)cc2)=O)c(N(C)C)ncnc1Cl C1(CC(=O)NC2C(CCOC)C2)CN(C(=O)C(C)n2cccn2)CCO1 CC(C)C(O)C(C)C(=O)NCCCCCC(=O)NCCC1CCCCCC1 c1(C(N2CC(N(C(C(N3CCN(C)CC3)C)=O)C)C2)=O)ccnc(Cl)c1 N1(C(C2C(C(C)C)(CC)C2)=O)CCC(CNC(=O)Cc2cc(COC)cs2)C1 C1(NC(c2ccc(O)nn2)=O)CCN(C(c2cnc(Cl)[nH]2)=O)CCC1CO N1(C(C(C(C)C)F)=O)CC(CNC(c2ccc3nn[nH]c3c2)=O)OC2CCCC12 Cc1sc(C)c(C(=O)NCC2C(C)CCCN2C(=O)C2CC2)c1Br CC1(NC(c2cccc(N(C)C)c2)=O)CCN(C(=O)Cn2cccn2)CC1 Cc1c(CNc2nc(N3CCCC3)cc(N)n2)ccc(Cl)c1Cl C(=O)(C(CNC(C1(C#C)CCCC1)=O)CC(C)C)N1C(C#C)CCC1 c1(C(N(C2CCCCC2C)CC(=O)OCC)=O)c(Cl)cc(Cl)c2ncccc12 CC1CN(C(c2cncc(N)c2)=O)CCCN1C(=O)CCC(C)(C)F c1(COC)cc(C(c2nnnn2CCCF)NC(C)CSc2cccnc2)no1 Cn1nc(I)cc1C(=O)NCCc1csc(C2CCS(=O)(=O)C2)n1 c1(CNC(CS(N)(=O)=O)=O)cc(O)nc(CNC(=O)CN2CCCC2=O)n1 c1(C(N(C(C)C)CCNC(C2CCSC2)=O)=O)ccc(CO)c(F)c1 c1(C(N2CC(C)CC(NC(CS(=O)(=O)NC)=O)C2)=O)cc2c(Cl)nccc2o1 c1(CN(CC)CC2CCOC2)ccc(OC)c(Br)c1 CC1CN(C(=O)C2=CCN(C(c3nc(=N)cc[nH]3)=O)CC2)Cc2nncn21 c1(C(=O)NCC2CCC(NC(CC3OCC(C)(C)C3)=O)C2)cc(N)c(F)cc1F c1(OC)cc(C(=O)NCCN(C(C2(F)CCCC2)=O)Cc2ccccc2)ncn1 N1(C(CC(C)SC)=O)CCCC2(CNC(c3cnc4c(c3)CCC4)=O)CCCC12 C1(C)(CC(NOCC(=C)Cl)=O)CCN(C(=O)C(CC)OCC)C1 c1(C(C2CC2)OC)nc(C(c2ccc(C)cc2)C)n(-c2nc(Br)nn2C)n1 N1(C(CC(CC)C2CCC2)=O)CCN(C(=O)C(C)OCOC)CC(O)C1 C1(NC(CCNC(C2C(C)C2)=O)=O)CC2CCC(C1)N2C(C12CSC(C1)C2)=O C(=O)(C(C)C(O)C(C)C)N1CCC(NC(c2c(C)nncc2)=O)C1(C)C Cc1cccc(C(N2CCOCC2C#N)C(=O)NCc2ccco2)c1I O=C1CCC(CNC(=O)COC2CN(C(=O)CCC3CCC3)C2)N1 C(=O)(C#CC1CCCCO1)NCc1nnc(CC)s1 c1(-c2ccc(N(C)C)cc2)n[nH]c(=Nc2cccc(F)c2CO)o1 C1(C(=O)NCCCNC(Cn2cccc(C)c2=O)=O)CCC2CCC(=O)N12 c1(CC(=O)NCC2CC(NC(c3cnc(O)o3)=O)CC2O)cc(F)cc(Cl)c1 c1(C(=O)NC2CCN(C(CC(=C=C)C)=O)CC(O)C2)cccc2c1OCC2(C)C c1(OC)cc(C(=O)NC2CC(C)(NC(=O)C(C3CCC(=O)N3)C)C2)cc(Cl)n1 c1(C(c2ccccc2F)(F)NC(N2CCCC(c3nnco3)C2)=O)cccc(F)c1 CCC(C)(C)C(C)CC(=O)NC1(C)CCN(C(C2CC(n3cccn3)C2)=O)CC1 c1(NC(C2CC(NC(c3ccc(O)c(Cl)c3)=O)C2)=O)ncc(O)cc1Cl n1(CC(=O)N(C(C)C)COC2CCOC2)cc(-c2cnn(C3CCCC3)c2)nn1 c1(-n2cc(CCC(=O)N(C(CC)C(=O)O)C)nn2)cc(OC)cc(OC)c1 CC1CC(C(=O)NC(C)(C)CNC(c2ccnc(N(C3CCCC3)C)c2)=O)=NO1 c1(C(=O)NC2CC(C)N(C(=O)C=Cc3ncc[nH]3)CC2)ccc2ccccc2c1 Cc1ccc(CC(=O)NC2(CNC(C3CC(C)(F)C3)=O)CCOC2)cc1[N+](=O)[O-] N1(C(CCN(C(C)=O)C)=O)CCCC2CCN(C(=O)Cc3ccc(O)cn3)CC12 C1(NC(C2(OC)CCSC2)=O)CCN(C(=O)C=Cc2ccncc2C)CC(O)C1 c1(OC)ncc(C(N2CCCC2CNC(=O)C(=Cc2cnc[nH]2)C)=O)cc1C C(=O)(CC(C)(C)C(F)(F)F)N(C1CCCN(C(C(CC2CC2)OC)=O)CC1)C Cc1ccc(C(=O)NCCCC(C)(C)NC(=O)Cn2cc(Cl)cn2)c([N+](=O)[O-])c1 CC(C)C(CCN(C(=O)C(C1CC1)C1CC1)C)NC(c1csc(Cl)n1)=O c1(OCC(=O)NCC(CC)NC(c2cnc(C(=O)NC)nc2)=O)ccc(F)nc1 c1(OC)cnc(Cl)c(C(N2CC(F)(C(=O)Nc3ccc(C(C)C)cc3Br)C2)=O)c1 C1(NC(CC(C)c2ccco2)=O)COCCC1NC(=O)CCc1nnc[nH]1 N1(CCNC(=O)C2=CCC2)CCCN(C(=O)CCn2cccn2)CC1 C1(C)(CNC(CN(C(COC)=O)C)=O)CCN(C(C2CCOCC2(C)C)=O)CC1 Cn1nc([N+](=O)[O-])cc1C(N1CCCC(F)(CNC(c2cc(=O)n(C)o2)=O)C1)=O C1(C)(C(=O)NCCCC(=O)NCC(CC)CC)CCC(C)CC1 C1(NC(C(C)C2CCCC2)=O)CN(C(C2CC23CCC3)=O)Cc2nccn2C1 C1(C2CC2)(NC(C2OCCN(C)C2)=O)CCN(C(=O)CC(C)(F)F)C1 C(CCC(C)C(=O)NCC=CCNC(c1n[nH]c(C)c1O)=O)OC N1(Cc2c(OC)c(F)cc(F)c2)Cc2ccccc2C1C(=O)N1CCCOCC1 C=CCCC(F)(F)C(=O)N1CCC(C(C)NC(c2ccccc2Cl)=O)C1 N1(C(CCn2ncc(C)c2)=O)CC2CCC(C1)N2c1ccc([N+](=O)[O-])cc1 c1(OCCCNC(C(C)OCC=C)=O)ccccc1OC(F)(F)F C12(C(=O)NC3C(NC(=O)CCc4ccnc(Cl)c4)COC3)COCC1C2(F)F C=Cc1cncc(C(=O)NCC(C)(O)CNC(=O)C(=Cc2ccco2)C)c1 N1(C(C2(C(C)C)CC2)=O)CC(NC(c2cnn3cccnc23)=O)C(N=[N+]=[N-])C1 C=C=CCC(C(=O)NC(C)CNC(c1ocnc1CC)=O)NC(=O)OC(C)(C)C C(CNC(c1cn(C2CC2)nc1C)=O)(CC)(CC)NC(C=CC=CCC)=O C(=O)(C1=CC2(CCOC2)C1)NC(CNC(C1=C(C)OCCS1)=O)CC(C)C C1(F)(CNC(c2nc(C)oc2)=O)CCN(C(c2ncccc2Br)=O)CC1 Cc1cc(=NCC(C)(C)C2=CCCC2)[nH]c(N2CC(C)OC(C)(C)C2)n1 n1(CCC=C)cc(C(=O)NCCN(C(=O)CC2CC=CCC2)CC2CC2)nn1 CC1(C)CCN(C(=O)CN(C(c2cc(C3CC3)on2)=O)CC2CC2)CC1 N1(C(C2CN(C3CCOC3)C2)=O)CCC(Nc2cc(C(N)=O)ncn2)CC1 c1(OC)ccc(C(N2CCOCC2CN(C)C(C2CC2(C)Br)=O)=O)cc1O c1(C(=O)NC(C)C(c2ccccc2)NC(C2CSCCS2)C)cnc(CO)cn1 CC1CN(C(c2cn(C)nc2Br)=O)CC(C)CN1C(c1ccnc(S)c1)=O Cc1nccc(C(=O)NC2(CNC(=O)C(C)N(C)C)CC2)c1N C1(CC(=O)NCC#N)CCN(CCc2ccccc2)C1 N1(C(c2cc(OC)ns2)=O)CCN(C)CC1C(=O)N(C1CCOC(C)C1)C Cc1cc(C(=O)N(C)CC2(O)CN(C(c3cccnc3C)=O)C2)c(O)nc1C C1(CC)(CNC(c2nnnn2CCSC)(C)CC2CC2)CCCCO1 N1(C(C2C(C)=CCS2)=O)CC(C(=O)NCC2CCCNC2=O)CCC1(C)C c1(C(=O)NC(CC)C2CCC2)ccc(S(=O)(=O)N(C)CC)cc1 C1(C(=O)NCC(CNC(c2ccc(NC)cc2)=O)OC)CS(=O)(=O)CCO1 c1(C(=O)NC2CC(NC(C(=O)OCC)=O)C2)ccc(S(=O)(=O)CC)cc1 n1(CC)ncc(Cl)c1C(=O)NC1(CNC(c2ccn(CC(F)(F)F)n2)=O)CCC1 N1(C(C2C(CCOC)C2)=O)C2CCC(C2)C1C(=O)N(C1CCCC1)C C1(C(=O)NC2CCC(NC(=O)CCOC3CCOCC3)C2)CCS(=O)CC1 C1(C(=O)NC(C=C)(C)CC)CN(C(=O)CC2COCC(C)O2)CC1N(C)C Cc1nn(C)cc1CC(=O)NC(C)CCC(=O)NCC1CCCOCC1 C(=O)(C1=CC2CC(C1)CC2O)NCC1(F)CC(CNC(Cc2ccc(C)o2)=O)C1 Cc1cn2nc(N3CCOCC(NC(C45CC(C)(C4)OC5C)=O)C3)sc2n1 N1(C(c2c(C)nncc2)=O)CCN(C(=O)Cn2cnc(C(F)(F)F)n2)C(CO)C1 C(=O)(C1=CC2CCC1C2)NCC1(OC)CCN(C(c2ocnc2C)=O)CC1 C1(CNC(C2CC(CF)C2)=O)CCN(C(=O)Cc2csc(Br)c2)CC1O C(=O)(C#CC1(C)CCCO1)NCC1C(C)(C)N(C(C2C3CCC(=O)C23)=O)CC1 N#CC1CN(C(=O)COC2CCCC2)CCN1C(=O)CCn1cncn1 C(C(=O)NCC1(C)CCCC1NC(C1CSCN1CC)=O)(C(C)C)OCCC CCN=C(NCC1(S(=O)(=O)N(C)C)CCC1)N1CCC(C(=O)NC(C)(C)C)C1 N1(C(CSc2n(CCC)c3c(n2)cccc3)=O)CCOC2(CCS(=O)(=O)C2)C1 C1(C(=O)NC2CCCC(NC(=O)CN3CC4CC4C3)C2)Cc2nncn2C1 N1(C(COCC(=O)NC)=O)CCC(O)(CCNC(c2cccc(F)c2C)=O)CC1 c1(SCC(C(=O)NCC(C)(C)OC)C)ccc(C(=O)OC)cc1Br N1(C(C2(CC#C)CCC2)=O)CCC(O)(CN(C(=O)Cc2nonc2C)C)C1 C12(C(=O)NC3C(CO)CCN(C(CC=CC=C)=O)C3)CC3CC(C1)CC(O)(C3)C2 CCCC(C)(O)CNC(C1(CC)CCN(C(=O)COC2CC2)C1)=O C1(NC(c2c(O)cccc2F)=O)COCCN(C(=O)Cc2ccc(Cl)c(F)c2)C1 c1(C(=O)NC(CNC(CCC(C)OCC)=O)CO)c(OC)cccc1O CC(CCCCNC(=O)C(C)(C)F)NC(=O)C(C)Oc1ccccc1.C1(O)CCCC1 c1(CCNC(N(C(CC)CC)C)=O)c(OC)ccc2ccccc12 CC1(NC(N2CCN(c3cc(C4CCCCC4)ncn3)CC2)=O)CCC(F)(F)C1 c1(-c2cnc(CCC(N3CC(C)(C(=O)NC4CC4CF)C3)=O)o2)ccc(F)cc1 Cc1cccc(CC(N2CCC(CN(C)C(c3ccns3)=O)C2)=O)c1 C(=O)(CC(C)C(C)C(C)C)N(CCN(C(C1CC2(C1)CC(OCC)C2)=O)CC)CC CCC(C)C(C(=O)NC1CCCC(NC(=O)C2=COCCO2)C1)SC N1(c2nnc(CC(C)C)s2)CC(NC(=O)C=CCF)C(C)C1 Cc1ccccc1CNC(=O)C(CCF)NC(C1(CC2CC2)CCC1)=O C1(C(=O)Nc2cnc(OC)nc2)CN(C(C2CC3(C2)CC3(F)F)=O)C2(CCC2)C1 c1(C(N(C2CCN(c3cc(-c4ccccc4)ncn3)C2)C)=O)cc(Cl)cn1C c1(C(N2CCC(CN(C(C(C)OCC)=O)C)C2)=O)cc(Br)cnc1N C(=O)(C(F)(F)C1(OC)CCC1)NCCN(C(=O)C(C)O)CCC C(=O)(CCC(C)NC(=O)CC(C)n1cccn1)N(c1cccc(F)c1)CC N1(CC(=O)NCCOCCNC(C2C(c3n(C)ncc3)C2)=O)CCC(=O)NC1=O c1(C(N2CCC(N(C(C3CC(O)C3)=O)CC)C2)=O)cc(C)c(F)cc1F c1(CC2(C(N3CCC(C(=O)NCC4CCNC4=O)C3)=O)CC2)cccc(Cl)c1 C(C(=O)N1CCC(C(=O)NCCCCS(C)=O)O1)n1ccc(C)n1 c1(CNC(C(C)OC)(C)c2nnnn2C(C)C)cc(F)c(Cl)cc1Cl Cc1cc(C(=O)NCCC(C)NC(c2cccc(F)c2C(F)F)=O)c(N)c(F)c1 C1(CC)CCN(C(c2cncc(O)c2)=O)C1C(=O)NOCC1CCCO1 C1(NC(C2(C)CC2(F)F)=O)CC2CCC1N(C(c1ccc(OCCF)cc1)=O)C2 CCC(O)C(C)C(=O)N1CCC(CO)(NC(=O)Cn2cc(C(F)F)cn2)C1 CC1CCC(NC(c2csc(C(F)(F)F)c2)=O)CN1C(C1CN(C)C(=O)N1)=O C1(CC#C)(NC(C2COCCC2NC(=O)C(=O)N(C)C)=O)CCCCC1 Cc1cc(C(=O)NCCCC(O)C(=O)N(C)Cc2ccn(C)n2)ncc1N c1(NC(CN2CCC(C#CC)C2)=O)cc(O)c(C)cc1C C=CC(C)(C)C(=O)NC1CC(C)N(C(=O)C(c2cccc(C)c2)=O)C1 C1(CC(N2CC(CC(=O)N(CC(F)Cl)C)(N(C)C)C2)=O)CC2C=CC1C2 N1(C(C2CCC(CC)O2)=O)CCC(c2cn(CCCOC)nn2)C1CC Cn1c(C(N2CC(NC(=O)C=CC(C)(C)C)C3CCCC23)=O)cc2occc12 C1(NC(C(C=C=C)C)=O)CCN(C(C2(Cl)CCCCC2)=O)CC1F C1(N(C)C(c2coc(Br)n2)=O)CCCCC1NC(C1(CCO)CC1)=O c1(COC)ccnc(-n2ccnc2)c1.C1C(NC(=O)OC(C)(C)C)CNC(=O)N1 c1(NC(N(CCCN2CCCC2)CC)=O)c(Cl)cccc1[N+](=O)[O-] c1(C(=O)NCC(CCNC(C(=O)NCC(F)F)=O)O)ccc2ccccc2c1F Cc1ccc(Cl)c(O)c1C(=O)NCC(O)CN(C(=O)CC=CC(C)(C)C)C c1(N(C)C)nc2ccc(C(=O)NC3CCN(C(c4cccc[n+]4[O-])=O)C3)cc2[nH]1 O=c1c2ccnn2cnn1CCc1ncc(C(F)(F)F)cc1Cl N1(C(C2(COC)CCC2)=O)CCCCC(CNC(=O)CCCCCO)C1 c1(C(N(CC(C)NC(CCOCCOC)=O)C)=O)cc2c(C)c(C)ccc2[nH]1 c1(C(=O)NC2C=CC(CNC(C(C)(C)CO)=O)C2)cnc2ccccn12 C(=O)(CC1=Cc2ccccc2C1)N1CCCC(N(C(=O)CC2(C)CC2(Cl)Cl)C)C1 C=CCC(F)(F)C(=O)NC(C)CCN(C(=O)COc1ccc(C#N)cc1)C c1(C(=O)NC(Cc2cccc(CC=C)c2)C(=O)OC)nc(C)n2c1CCCC2 c1(C(N2CCN(C(C(C)=C(CC)C)=O)C(C(F)F)C2)=O)cnn2c1CC(C)CC2 N1(C(C2C(C)CCCC2)=O)CC2CC(C(=O)NCCC3(C)CC3)(C2)C1 c1(C(=O)NCC2CN(C(CCNC(COC)=O)=O)C(C)C2)c(F)cc(F)c(F)c1F N1(C(CC(C)F)=O)CC(C)(C)CC1CNC(C12CCC(CO)(CC1)C2)=O S(=O)(=O)(c1cccc(Cl)c1)N1C(C(=O)Nc2cnc(Cl)c(Br)c2)CC(F)C1 C1(C(N2CC(NC(c3c(OC)nc(Cl)cc3)=O)C2)=O)CCC2CC(C)CN2C1 C(=O)(CC(=O)N(CC(O)CN(C)C(C1(CCC)CCC1)=O)C)NCC#C c1(NC(CC2CC(=O)NC2)=O)nc2c(s1)CC(c1ccccc1)CC2 c1(C(N2CCCC2CCC(C)C)C(=O)NC(C(=O)OCC)C)ncc(Cl)cc1Cl C1(C(=O)NC(C)CCO)CCN(C(C2CC3(CCO2)CC3)=O)C12CCC2 C1(NC(=O)NCCOC)CCC(CCNC(=O)Nc2cccs2)C1 c1(CCC)ncc(C(=O)NCC2CCCC2NC(=O)C(C)CO)s1 c1(OC)ccc2nc(C(=O)NC3CN(C(C4CC4F)=O)CC3(F)F)ccc2c1 C1(C(N(CCCNC(c2ccc(C)s2)=O)C2CC2)=O)CC12CC(F)(F)C2 N1(C(CC2ON=C(C)C2)=O)CCC2CCCC12C(=O)NCC1CCOC1C C(CC(=O)NCCN(C1CC1)CC)N(C(=O)CC1CC1C(F)(F)F)CC C1(NC(c2scc(-c3cc(C)ncc3)n2)=O)CCc2ccccc2C1 C(C(C(=O)NCCCCc1ncc[nH]1)C(C)C)NC(c1cc(C(C)=O)on1)=O c1(C(N2C(CNC(C(CCC)OCC)=O)CCC2)=O)cnn(C)c1C#N N1(C(CCC2C(C)=NNC2=O)=O)CCC2(CC1)CN(C(c1ncsc1C)=O)C2 c1(C(N2CCC(CNC(C3(F)CCCC3)=O)C23CC3)=O)cc(Cl)cc2c1OCC2 C(c1ccc2c(c1)OCO2)=CC(=O)NCC1(NC(C2CCSC2)=O)CCC1 N1(C(C(c2cc(C)cc(F)c2)C)=O)CC2(C)CN(C(=O)C(C)C(C)O)CC2(C)C1 CC1c2c[nH]nc2CCC1C(=O)NC12CC(CNC(=O)CC3CCCOC3)(C1)C2 Cc1ccc(-c2ocnc2C(=O)NC(C)CNC(C2C(C)(C)C2(F)F)=O)cc1 c1(C(N2CCC(N(C(c3ccccc3)=O)CC)CC2)=O)ccc2oc(O)nc2n1 Cc1cncc(N(C(COC)=O)CC(C)CCN(C(=O)CC2CCCC2O)C)n1 C1(OC)CN(C(=O)CNC(=O)NC2CC2)CC1NC(c1cccc(N)c1)=O N1(C(C(CC)=CC)=O)CCN(C)C(C(=O)NCCN2CC3CCC2C3)C1 C1(NC(C(COC)C)=O)CC2(CCN(C(c3nnccc3C)=O)CC2)C1 CC(C)(C)CC(C)(C)C(=O)N1CCOCC(NC(C2CCC=CCCC2)=O)C1 N1(C(C(C)CC2CC2)=O)CCC(NC(=O)CNC(c2ccco2)=O)C(CO)C1 C(=O)(CC(C)(C)C(C)(F)F)NC1CCN(C(C2N(CC)CCOC2)=O)CC1(F)F N1(C(C(CC)(C)C(=O)OC)=O)CC2CCN(C(=O)Cn3nccn3)CC2C1 C1(C(N2C(CNC(c3c(C)nccn3)=O)C=CC2)=O)CCc2ccccc2C1 C(=O)(CC(O)CCCCC)NCC(CC=C)NC(C1(CC#C)CCCC1)=O C1(NC(=O)COC(c2cccc(C3(O)COC3)c2)=O)CCCC(=O)N1 CC(C)(C)C(CS(C)(=O)=O)NC(c1nc(N2CCOCC2)ncc1Cl)=O N(C(=NCCS(C)(=O)=O)NCCS(=O)(=O)NC(c1ccccc1)C)C(CC)C C1(C(=O)NCC2C(CNC(c3c(CC)c(C)sc3)=O)C2)CCC2(CCOC2)O1 Cc1cc(C(=O)NC2C=CCN(C(c3ccc(O)nc3Cl)=O)C2)cc(=O)n1C C1(F)(C(=O)NC(C2CCOCC2)C#C)CCCN(C(c2cn(C)cc2C)=O)C1 N1(C(C(CCC)N(C)C)=O)CCC2(CC1)CC2C(N1CCn2nccc2C1)=O C(=O)(CC(C)(C)CC(=O)N1CCN(C(c2n[nH]cc2Cl)=O)CC(C)(F)C1)OCC C1(C(=O)OC(C)(C)C)CC(S(C)(=O)=NS(=O)(=O)c2cccc(OC(F)(F)F)c2)C1 Cc1cc(Cl)ccc1OCC(=O)NC1CCCC1CNC(C1CC2(CCC2)C1)=O c1(C(NNC(=O)Nc2c(C)n[nH]c2)=O)cc([N+](=O)[O-])c(C)cc1Br N1(C(COc2cc(C)on2)=O)CCCN(C(c2ccnc(C(N)=O)c2)=O)CCC1 C#Cc1cc(F)cnc1NC(C1CC1NC(=O)OCCc1ccccc1NC)=O C(=O)(C1=C(Cl)CCCC1)NC(CC(=O)NC(C)CC(C)(C)C)C(F)F C1(C(=O)NCC(C)F)CCN(C(=O)CC(C)CN(C)C)C1C C#CCC(C)(C)C(=O)NCC1CCCCN1C(C)=O C(=O)(C(C)(C)COc1cnn[nH]1)NCC1(NC(c2nc(OCC)oc2)=O)CCC1 C1(CC(N2CC3C(CN(C)C(C4(C)CC4)=O)C3C2)=O)CCCCC(=O)N1 C1(NC(C(CC)O)=O)C=CCCC1C(=O)NCCc1cn(C)nn1 C(c1cncnc1O)=CC(=O)NCC1N(C(C(COC)O)=O)CCOC1 CC(C)C(C(=O)NC(CNC(c1cncc(C(F)F)c1)=O)C1CCC1)NC(N)=O Cc1nc(C(=O)NCC(C)CN(C(=O)C(C)C2CC2)C)cc(O)n1 N1(C(C(F)=CCC)=O)CCN(C(c2nc(C)ccc2F)=O)C(CCO)C1 CC1C(NC(=O)C(=O)NCC2CC2)CC2CCC1N2C(C1(O)CCSC1)=O C(=O)(C(O)CCNC(=O)C(CN(C)C)NC(=O)CC1CC(=O)C1)OC c1(C(N2C(CNC(c3cc(C)oc3C)=O)CC(C)(C)C2)=O)cc(F)c(O)c(Cl)c1 CC(C)CCC(CO)NC(=O)CN(C(=O)C(C)CC1CC1)C c1(OC)cc(CN(C)C(C2(NC(=O)C=Cc3nccs3)CCC2)=O)on1 c1(C(=O)NCCNC(=O)CC2CC3CC3C2)ccc2c(c1)C(=O)NCC(=O)N2 c1(C(N(CC(O)CNC(=O)CC2COC(C)(C)C2)C)=O)ccc(Cl)cc1F C12(NC(CC=C=C)=O)CC3CCC(C1C2)N3C(=O)C(C)Cc1ccc(F)cc1 C1(C(=O)NCCCC2(NC(OC(=N)O)=O)CC2)CC(CCC2CC2)C1 C1(C)(CNC(c2scc(OC)c2)=O)CCN(C(=O)Cn2nnc(=O)[nH]2)CC1 C1(C(N(C2CCCN(C(=O)Cc3cccnc3)CC2)C)=O)CC2(C1)CC2(F)F C#CC1(O)CC(C(=O)N(CCNC(=O)CSCC(F)F)CCOC)C1 N1(C(CCNC(C=CCOCCOC)=O)=O)CCC(C)(CN(C)C)C1 N1(C(CCC=CC(C)C)=O)CCC2(CC1)CC2NC(=O)CSCC1CCCO1 N1(C(C2CCCN(CC)C2)=O)CC2=C(C1)CN(C(=O)CCn1ccnc1)C2 C(=O)(C1CCCc2ccccc21)NCC(CC)NC(c1cc(C#N)ccc1N)=O Cc1ccnc(CNC(c2nnnn2CCN(C)C)C2CCCCO2)c1Br c1(C(=O)NCCOC2CCN(C(C=CCCC(C)C)=O)CC2)ccc(=O)n(C)n1 C1(OC)(CNC(Cc2ccccc2)CO)CCNCC1 Cc1ccc(C(=O)NC2CC2NC(=O)C(C(C)C)c2ccccc2)c2c1CCC2 c1(OC)cc(N)cc(C#N)n1.c12ccc([nH]1)C(=O)C(=O)CC2.C(CCO)NCCCO N1(C(CC(CC)(F)F)=O)CC(NC(=O)CCCc2cncs2)CC12CCCCC2 CCC(C)C(O)C(C)C(=O)N1CC(C)(NC(c2cc3cccnc3[nH]2)=O)C1 N1(C(C2CCN(C)CC2)=O)CC2(CC2)CC1C(=O)NC(c1ccc(Cl)cc1)CO C1(CC#C)(C(=O)NC2CCC2NC(C2CC3CC2C3)=O)CC=CCC1 CC(C)(CC(F)F)C(=O)N1CC(CNC(C2CNC(=O)C2)=O)C(O)C1 CCCCC(O)C(=O)NCC1(COC)CCN(C(=O)CNC(N)=O)C1 C1(NC(C2(OCC)CCCC2)=O)CC2CCC1CC2NC(c1cnnc(C)c1)=O c1(C(N2C3CC4(NC(CCC=C)=O)C(C2CC3)C4)=O)ccnc2ccc(O)cc12 N1(C(C2C(=C)C2)=O)CCC(NC(=O)CC(C)(C)c2ccccc2)C(C)C1 C(=O)(CCS(C)(=O)=O)NC(CN(C(=O)CCOc1cccnc1)CC)C CCCC(CC)CCC(=O)NC(CNC(c1cnc2nc(C)oc2c1)=O)CC N1(C(C2(NC(c3cc(C)c(O)nc3)=O)CCOCC2)=O)CC(CO)CC(C)(C)C1 N1(C(C2(SC)CCC2)=O)CCOCC(F)(CNC(c2cn3c(n2)COCC3)=O)C1 N1(C(C2CC(=C)C2)=O)CC2CCC1C(CNC(=O)CC1COC3(CCC3)CO1)C2 N1(C(CC2(C=C)CN(C(=O)C(C)(F)C(C)(C)F)C2)=O)CCn2c(C)cnc2C1 C1(CN(C)C(C2CC=CC2)=O)CCCN(C(=O)Cc2cn[nH]c2)C1 C1(C(=O)NC2CC(CNC(c3csc(Br)c3)=O)C2)CC(O)(C(F)F)C1 C12(C(=O)NC(c3ccc(Cl)cc3)C)CCC(C(N3CCCC(O)C3)=O)(CC1)CC2 c1(C(=O)NCC2(NC(CC3CC(SC)C3)=O)CCCC2)nccc(Cl)c1F Cn1cc(-c2ccc(C3CC3)c(F)c2)c2cc(Br)ccc12 N1(C(CC2(OC)CN(C(C3CCC4(CCC4)C3)=O)C2)=O)CCC(O)C(C)(C)C1 O=C1CCC2(C(=O)NCC3CCN(C(=O)COC4CC(F)(F)C4)C3)SCCN12 c1(NC(C2(C)N(C(C(CC)O)=O)CCC2)=O)ncc(Cl)cc1[N+](=O)[O-] N1(C(C2C(=C)C2)=O)CCC(CCOC)(NC(=O)CC2OCCC2C)CC1 Cc1ccc(C(=O)NC2(CNC(c3cc4oc(Br)cc4[nH]3)=O)CC2)c(F)c1Cl C1(C(=O)NCC2(C)CCC(NC(=O)CCc3ncc[nH]3)C2)CN2CCN1CC2 C=C1Cn2c(C(=O)NCC3CC(NC(c4nc(O)sc4C)=O)C(O)C3)nnc2S1 C(=O)(C#CC(C)(C)CNC(=O)CC1COCCOC1)NC(c1ccn(C)n1)C N1(C(CC(C)OC)=O)CC2(CCN(C(=O)Cc3cccc(O)c3)CC2)C1C(C)C C(c1ccc(C(N)=O)o1)=CC(=O)NC(CC)CNC(C12CC(C)C1C2)=O C(C(C)N=c1cc(Cl)c(O)n[nH]1)NC(CC(C)OC)=O c1(CNC(C(CNC(=O)Cn2[nH]cnc2=N)OC)=O)cccc(C)c1F Cc1ccnc2nc(C(N3CCC(NC(C4CCS(=O)(=O)N4)=O)C3(C)C)=O)nn12 c1(C(=O)NC(C2(O)CCN(C(c3cc(C)no3)=O)C2)C)ncn2ccccc12 C1(CNC(C(C)CN2CCCCC2)=O)CCCN(C(=O)C(O)CN(C)C)C1 c1(Nc2n(C)ccn2)cnc(CN2CCC(N3CCNCC3)CC2)nc1 c1(C2(C(N(CCNC(C(=O)NCC)=O)C)=O)CCC2)ccccc1F C1(N(C(CC(CN(C)C)(C)C)=O)C)CCN(C(=O)C(C)(C)C#N)CC12CC2 N1(CC#CC)CCC(NC(c2nccnc2C(N)=O)=O)C(C)C1 C1(CC(=O)NCC2CCC(=O)O2)CCCN(C(=O)C=Cc2cc[nH]n2)C1 c1(C(=O)NC2CN(C(CN3CC(C)C3)=O)CC3C2C3)ccc2nc(O)oc2c1 Cc1cn2[nH]c(=NCC3CN(C(C4CS(=O)(=O)C4)=O)C3)sc2n1 N1(C(C(CO)OC)=O)CCN(C(=O)COC2CCCCC2)CC1C1CCCC1 C1(O)(C(C)NC(C2CCC2CF)=O)CN(C(c2ccc(-c3cccnc3)s2)=O)C1 O(NC(=O)C1=CC2C=CC1C2)C(CC(C)C)C(=O)N1CCS(=N)(=O)CC1 C#CC1CCN(C(=O)C(C)CN(C(=O)Cc2ccn(C)c2)C)C1 c1(OC)ccc(C)nc1C(=O)NCC1CN(C)CCN1C(=O)C(CCSC)OC c1(NCc2ccc(CCNC(C3N(C)CCCC3)=O)cc2)cccc2c1OCO2 N1(c2nnc(COC)s2)CC2(CCC2)CC1CNC(C1CC2CCCC(C1)C2)=O C(=O)(C(C)(C)CC)N1CC(c2cn(C(C(=O)OCC)C)nn2)(O)C1 N1(C(c2c(C)cccc2)=O)CCN(C(=O)Cc2ncncc2Cl)C(C2CCC2)C1 N1(C(C(CC)C)=O)CC(NC(C2CC2c2ccc(F)nc2)=O)CC(F)C1 c1(OC)ccc(C(N2CCC(C)C2CNC(=O)C(C)OCC(F)(F)F)=O)cc1Cl C12(NC(c3cn(CCC4CC4)nn3)=O)CC1CN(C(=O)Cn1cc(Br)cn1)C2 C1(C(=O)NCCCCCCN(C)C(C2CCC3CC23)=O)Cc2ccccc2O1 N1(C(C(C(C)C)C2CCC2)=O)CCC(C(=O)NC(C)(C)CC2CCOC2)C(C)C1 C(CC(C(C)(C)C)NC(C1CC1(C)COC)=O)N(C(C(C=C)CC)=O)C CC1CN(C(=O)CCC(C)(C)NC(c2ccn(C)n2)=O)CCC1(F)F C1(C(=O)NCCOCC(C)C)(NC(C2CC(CC)C2)=O)CCN(C)C1 c1(OC(C)C)cc(NC(N2CCCOCC2C)=O)ccc1Br c1(CNC(NCC(=C)Cl)=NCCC)ccccc1[N+](=O)[O-] c1(CNC(=O)C2=CCCC2)ccc2c(c1)CCC2NC(C1CC2(CSC2)C1)=O C#CCCC(=O)NC(C)(CNC(c1coc(CO)c1)=O)CC c1(C(=O)N(CC(F)CNC(c2cccc[n+]2[O-])=O)CC)cc(=O)c2ccncc2o1 c1(COC)ccc(C(=O)NCC2CC(O)(CNC(c3cnc[nH]3)=O)C2)o1 C1(CNC(C(C=C)OC)=O)CC(C)CCN1C(=O)C(CCSC)OC N1(C(CN(C(C)=O)CO)=O)CCC2(CC1)CN(C(=O)CCc1c(C)n[nH]c1C)C2 N1(C(C2CC(=C)C2)=O)CCCCC1CN(C)C(c1nc(C)cs1)=O C1(C=O)COCC1NC(=O)NC(N)=O.N12CC(C1)N2C.C(C)(C)C C1(NC(C(CC)C(C)O)=O)CCN(C(=O)CCn2cncn2)CCC1CO c1(C(N2CC(OC(C)(C)C)CC3(C2)CC3)=O)ccc2ccccc2n1 c1(C(N2CCC(CN(C)C(c3sccc3Cl)=O)C2)=O)ncnc(O)c1F C=CCC(C)(C)C(=O)N1CC(NC(=O)C(C2CC(F)(F)C2)OC)CCC1C N(C1CCc2cc(OC)ccc21)CCC(CC)(C)Nc1ccc(C)c(OC)n1 c1(CC)noc(CC)c1CC(=O)NC(C1CCCN(C(=O)COC)C1)C c1(SC)ccc(CNC(C2(O)CCN(C(=O)CN3CCOCC3)C2)=O)cc1 N1(C(c2oc(C)c(CO)c2)=O)CCC(CNC(=O)CN2CCCC2)C(C)C1 C(=O)(C(F)CCC(C)C)N(C1CCN(C(CC2(OC)CCOCC2)=O)C1)CCO N1(C(C=COCC)=O)CCC2(CC1)CC(NC(=O)C(C)CC(C)=O)CO2 N1(C(CC2CC(C)CC(C)C2)=O)CCC(c2nn[nH]n2)C(F)(F)C1 C1(CNC(c2c(CC)nn(C)c2)=O)CN(C(C2(C)CCC(=O)N2)=O)CCC1C CCC(C(=O)OC)(c1ccccc1)NCC(C)(C)C1CC1 C1(NC(c2ocnc2C(F)(F)F)=O)CCCCN(C(=O)C=Cc2nccs2)C1 c1(C(=O)NC2CCC(CNC(C(CN(C)C)O)=O)CC2)ccc2c(ccn2C)c1 c1(C(N2CCN(C(Cc3cnc(C)[nH]3)=O)CC2C(F)F)=O)ncc(C#N)cc1Cl C(=O)(C#CC1(C)CCCO1)NCCCN(C(c1c(OC)ccc(C(F)F)c1)=O)C C(CCCCOC)(C(=O)NCc1cccc(Cl)c1)N(C(C(=O)OCC)C)C C(=O)(C1Cc2ccccc21)N(CCC(C(C)C)NC(c1c(C)nns1)=O)C C1(NC(C#CCNC(C2N(C)CCCC2)=O)=O)CCC2(CCCC2)C1 C1(C(=O)NCc2n(C(C)C)cnc2)CCC2CCC1N2C(c1cnnn1C)=O C(=O)(CC(O)(c1ccccc1)C1CC1)N(CC(CNC(CC(=O)NCC)=O)O)C N1(C(C(c2ccc(F)cc2)(C)O)=O)CCN(C(C23CC(CO)(C2)C3)=O)C(CO)C1 c1(CC)n[nH]cc1C(=O)NCC(CC)NC(c1cnc(-c2ccccc2)o1)=O C1(O)(CC)CCN(C(c2ccc(C)nc2O)C(=O)Nc2cccc(C)c2Br)CC1 c1(C(N2C(CNC(c3cccc(F)c3)=O)C3CC3C2)=O)cc(F)ccc1Br C1(CNC(=O)CNC(c2ccoc2)=O)CN(C(C2CCC=CCC2)=O)CC12CC2 c1(C(=O)NCC2C(CNC(C(CC(C)C)(C)O)=O)C2)cccc2nc(O)[nH]c12 C(N=c1[nH]c(N2CCC(F)(F)C(F)C2)nc2c(F)cccc12)c1ccc(C)s1 Cc1nc(O)sc1NC(=O)NC(C)C(=O)N(c1ccccc1)C C(=O)(C1=C(C)OCCS1)N1CCCC(NC(CCNC(C)=O)=O)C1C c1(C(N2CC(C(C(=O)N3CCC3C(C)C)OC)C2)=O)cc(C(N)=O)no1 c1(CC)cc(C(=O)NCCCN(C(=O)CCc2c(C)noc2Cl)C)nn1C c1(OC)cc(C(=O)O)ncc1NC(=O)Cc1nc(Sc2ccccc2)n[nH]1 CCCC(C(O)C(=O)NCC(CO)C(C)(C)C)NC(c1cnn(C)c1)=O C1(CNC(CCC(=C)Cl)=O)CC2(CCC2)CN1C(=O)C(C#N)C(C)(C)C c1(CC(=O)N(CCCN(C(=O)CNc2ncccn2)C)C)ccc(F)cc1 c1(C(=O)NCCC(C)N(C(C(=O)Nc2ccc(C)cc2)=O)C)ncc(Cl)cc1F c1(C(N(C(C(C2(N3CCOCC3)CCCCC2)C)=O)C)C)cccc([N+](=O)[O-])c1 c1(C(C)=O)cccc(-c2cn(CC(=O)NCC(=O)NC3CCS(=O)(=O)C3)nn2)c1 c1(C(=O)NCCC(C)N(C(=O)C(C)c2cccs2)C)cccc2c1CCC2=O c1(OC)cccc2c(C(=O)NC3CCCN(C(=O)C(Br)=C(C)C)C3)csc12 N1(C(C2(CCC=C)CCCC2)=O)CCCCC(NC(=O)CC2C(=O)NN=C2C)C1 N1(C(CCC(=C)Cl)=O)CCN(C(c2cc(C3CC3)nn2CC)=O)CC1CO c1(C(=O)NCC(C2CC2)NC(c2cnc(C(C)OC)s2)=O)cccc2nncn12 c1(C(=O)NCC(CNC(CC(C=C)c2ccccc2)=O)O)scc2c1CCCC2 c1(C(=O)NC(C(C)NC(=O)Cn2ncnn2)C)conc1C1(C)COC1 N1(C(C(C(C)C)NC(C2CCOC2)=O)=O)CCC(CN(C)C)C(C)C1 C1(NC(CSCC(C)C)=O)CN(C(=O)CCc2cn(C)cn2)C2(CCCOC2)C1 C1(C)(C(=O)NC2CCCN(C(C(C(C)(C)C)=O)=O)C2)CCCNS1(=O)=O C1(NC(COCCN(C)C)=O)CCC2CC1CN2C(C1CCCCC1O)=O c1(C(N2C(CNC(CC3CC(CC)C3)=O)CCC2)=O)cc(C)nc2ccccc12 C1(CCNC(=O)C(C)OCC(C)C)(OC)CN(C(c2ccsc2)=O)C1 C(CCCCC(=O)N1CCC2(CC2NC(C2CCC(=O)N2)=O)C1)OC C#Cc1cn(C)nc1C(=O)N(C)CC1(O)CCN(C(=O)CC2CCCC2C)CC1 C(=O)(CCC(C)N(C)C)NCC1C(C(=O)NC(CC=C)CO)CC1 C12(CCNC(=O)NCc3cc(C)cc(Br)c3)CC3CC(CC(C3)C1)C2 c1(C(N(C2(C(=O)NCC(C3CCCC3)OC)CCC2)CC2CC2)=O)cc[nH]c1C N1(C(C23CC(CC)(OC2)C3)=O)CCC(NC(C2CC3CCC(C2)C3)=O)C(C)C1 C1(O)(CN(C)C(C2CC(O)C2)=O)CCN(C(c2conc2C2CCCC2)=O)C1 C=CCC(C(=O)OC)NC(C1COC(CNC(=O)Nc2cn(C)nc2C)C1)=O C(C(CC(C)C)C(=O)NC(CC1ON=C(C)C1)C)NC(=O)CCCc1ccc(N)cc1 c1(C(N2CCCCC(NC(C(CC=C)(F)F)=O)C2)=O)cccc2nonc12 c1(C(=O)NC(C(=O)NC2CC3CC3C2)c2ccoc2)ccc(CO)nc1 C1(OC)CC(C(=O)NCCCN(C(=O)C=Cc2cscn2)C)CC1OC c1(CC(=O)N(C(C(=O)N(C(C)C(=O)OC)CC=C)C)C)ccc2c(c1)CC2 c1(CC(=O)NCC2N(C(CSCC(N)=O)=O)CC3CC32)cccc2nsnc12 C1(C(=O)NC(C(=O)NC2C(C)(C)C2(C)C)C2CCOC2)CC2(CCO1)CC2 c1(C(=O)NCC(CNC(=O)CC2CCOCC2)F)cnnc(-c2ccccc2)c1 CC1=NOC(CC(=O)NCC(C2CCC2)NC(C2CC(O)C2)=O)C1 c1(C(=O)NC2(C)CCN(C(c3c(COC)cc[nH]3)=O)C2)cccc2nn[nH]c12 C#CC1CCCN(Cn2nc(-c3cnccn3)n(CC)c2=S)C1 c1(C(COC)(C)C)n[nH]c(=NC2Cc3ccc(Br)cc3C2)o1 CCC(C(=O)N1CC(CNC(=O)COC(C)C)C1)n1cccn1 C(=O)(C1=NOC(CNC(c2c(C#N)cnn2C)=O)C1)Nc1c(C)n(C)nc1 Cc1cc(N2CCCC(NC(c3ccsc3Cl)=O)C2C)ncc1C#N C1(C(=O)NC)CCOC(C)(CC)C1.C#CCC1C(=O)NC2C(CC2)C(=O)N1 C1(NC(C(N2CCCCCC2)C)=O)(CNC(C2CCOC2=O)=O)CCCCC1 c1(C(=O)NC(C(=O)NC(CC)CCOC)Cc2cc[nH]n2)cc([N+](=O)[O-])n[nH]1 N1(C(c2c(COC)nn[nH]2)=O)CCCC2(C1)CN(C(=O)Cc1csc(Cl)n1)C2 C1(C(C)C(=O)N2CC(OC(=N)O)C2)CCN(C(=O)C=C2CCC2)C1 C1(N(C(C(C2CC2)SC)=O)C)CN(C(=O)C=Cc2cccs2)CCC1O CCCC(O)CC(=O)N1CC2C(c3cn(C(c4cc(C)cc(C)c4)C)nn3)C2C1 CCCC(C)(C)CC(=O)N(CCCCCC(=O)NCC(c1ccncc1)O)C C1(NC(CCC2CCN(C)C2)=O)CCCCCC1NC(=O)Cc1ccns1 N1(N(C2CC(C#N)C2)C)CC2(C1)CN(C=O)C2.C12(C=O)CC3CC1C2C3 [N-]=[N+]=NC1CC2(C(N3CCC(OCCNC(c4ccon4)=O)CC3)=O)CC12 C(N=c1[nH]c2c(c(=NCC3C4COCC34)[nH]1)CSC2)c1nccc(O)n1 C1(C(=O)NCCOCCNC(c2ccoc2)=O)CS(=O)(=O)CC1c1ccccc1 C(=O)(CCCC(C)(C)CC)NCC1CC(O)(CNC(C2(C(=O)NC)CC2)=O)C1 N1(C(C)C)C2CCC1CC(NC(C1(CNC(=O)C3=C(Cl)CC3)CC1)=O)C2 N1(C(C=COCC)=O)CC(C)N(C(=O)Cc2nnc(O)s2)CC1C c1(OC)cnc(SC)nc1N(C1CCNCC1F)C(c1cc(C(C)C)no1)=O Cc1cc(C)[nH]c(=NCc2ccc(Sc3c(F)cc(F)cc3F)s2)n1 c1(CC)ccc(C(=O)NC2CCN(C(=O)C(O)COC)C2(C)C)cc1CC C#CC1CCCN(C(C2CCC(Cn3cc(CC4CCCN4C)nn3)CC2)=O)C1 C1(C(=O)NC2C(CNC(CCOCCC)=O)COC2)COc2cc(Cl)ccc2C1 Cc1ccc(F)c(C(=O)NCCC2(C)CCN(C(C3CCCC(=O)N3)=O)C2)c1F CCCCCS(=O)(=O)CC(=O)NCC(CCNC(=O)Cn1ccc(C)n1)OC N1(C(CCCOC(C)=O)=O)CCC(C)C(NC(c2cc(F)cs2)=O)C1 c1(CC(C(=O)NC2CC(C)(NC(C=NOC)=O)C2)O)cccc(Cl)c1 c1(C(=O)NC2CN(C(=O)C=C3CC3)CC23CC3)ccc2nc3n(c2c1)CCC3 n1(CC)nc2c(c1C(=O)NCC1CN(C(=O)CCCN=[N+]=[N-])CC1O)CCCC2 c1(N(C(c2ncc(-c3ccc(F)cc3F)o2)C)C)nc2c(c(=N)[nH]1)CCCC2 N1(C(CS(=O)(=O)NC)=O)CCOC2(CCN(C(C3CC(C(=O)OC)C3)=O)C2)C1 C1(NC(C(C)C2CCC2)=O)COC2(CCN(C(=O)Cc3ccc(F)cc3)CC2)C1 C1(NC(C(c2n(C)cnc2)=O)=O)CC2CC(C1)N(C(=O)CCC1(C#N)CCC1)C2 C#Cc1ccc(C(=O)N(CC(=O)NCCCS(C)=O)CC)cn1 C(CCCC(=O)NC1CCN(C(c2cccc(C)n2)=O)C1C1CC1)OCC C1(CNC(CCC2CCN(C(c3c(CC)cccc3)=O)C2)=O)CC2CC1CC2O C(=O)(C(CNC(=O)C(C)(C1CC1)OC)CC=C)NC(C#C)C1CCC1 N#Cc1ccsc1C(=O)NCC1(F)CC(NC(C2CCCC(C3CC3)O2)=O)C1 C1(COC)CCCN1C(C1(CCl)CN(C(C2CC2c2cccs2)=O)C1)=O CC(C)(C)CCCC(C(=O)NC1CCOC1)N1CCOC(c2ccco2)C1 C12(C(N3C(C)CC(C)(C)C3)=O)CCCC1CN(C(c1ccc(CO)o1)=O)C2 C1(C(N2CC(CC(C(=O)N(CCO)C(C3CC3)C3CC3)F)C2)=O)CCCC12CCC2 S(=O)(=O)(c1cc(C(=O)OC)c(Br)cc1F)N1CCCN(CCOC)CC1 N1(C(c2c(C)n(CCC#N)nc2)=O)CC(C2(NC(c3ccc(Cl)cc3)=O)CC2)C1 C(=O)(CCCCN=[N+]=[N-])NCC1C(C)(C)C1C(=O)NCC1(O)CCCOC1 CC(C)CCCCCC(=O)NC1CCN(C(C2CC3(CCCC3)C2)=O)C12CC2 C12(C(=O)NCCCNC(c3cccn3C3CC3)=O)CCCC(=O)N1CCC2 CCCCC(C)C(=O)NCCC1CN(C(C2CC(CC(F)F)C2)=O)CCCO1 C1(CNC(C2(CNC(C(C)OCOC)=O)CC=CC2)=O)OCCCC1(C)C c1(C(=O)OCCC2CCCC23CC3)nc(C(F)(F)F)oc1Br N1(C(C(CC)F)=O)CC2(CCN(C(C3CCSC3)=O)C2)C1 CC1=C(C(=O)NC(CNC(=O)C(=O)NCCSC(C)C)CO)CCC1 CC(C)C(O)C(=O)NCC1C(CO)CCN1C(=O)C=Cc1ccn(C)c1 C1(CNC(C2C(C=C)CC2)=O)CC(F)(F)CN1C(=O)CCc1nnc(O)nc1O c1(OC)ccc(NC(C2CCN2C(c2ccc(-c3cccs3)[nH]2)=O)=O)cc1C#N N1(C(C(CC(C)C)C)=O)CCOC2CN(C(c3cnc4n3CCCCC4)=O)CC12 C1(C(=O)NCCC2(COC)CC2)C=CCN(C(c2ccn(C3CC3)n2)=O)C1 N1(C(CCSCC)=O)CCCCC1C(=O)N(C1CCOCC1C)C C(=O)(CCC(=O)NC1COCC1NC(=O)C(Cl)=CCl)Nc1nnc(CC)s1 Cc1occ(C(F)(F)F)c1C(C)NCCN(c1nnnn1C)C(=O)CO CCCCC(CC)C(=O)N1CCC(CCNC(C2C3CCN2CC3)=O)CC1 c1(OCC)c(NC(c2ccccc2)c2ccccc2)cccc1C#N C(=O)(CCCC(C)(C)NC(=O)C(F)=CC1CC1)NCCC1(C)CCOC1 C(=O)(NNC(=O)NCc1cccs1)NC(CC)Cc1nn[nH]n1 N12CCC3(CC1)CC(C)N(C3)C(=O)C1C(C1)C2=O.C1(COC)CC(OC)C1 C(=O)(CCC1CCc2ccccc21)NC1C(C)CN(c2nc(Cl)ncc2Cl)C1 c1(C(=O)NCCN(C(=O)CCn2cnc([N+](=O)[O-])c2)CC)cc2c(o1)CCCC2 C1(NC(=O)CN2CCOCC2=O)(CO)CCCN(C(=O)CCCCC2CC2)C1 c1(C(=O)NC(CCOC)CNC(c2nnn3c2CCC3)=O)n[nH]c2c1CCCC2 N1(C(c2c(C)nn(C(C)C)c2C)=O)C2CCC1CN(C(c1cccnc1C)=O)C2 N12CCCC(C)(C1)NC(=O)c1ccc(o1)C2=O.C1C2COCC12.N(CC)(CC)C C(=O)(C1CCc2ccccc21)N1CCCCC(C(N(c2cnn(C)c2Cl)C)=O)C1 N1(C(C2CCCN2c2ccncn2)=O)CCC(F)(c2ccccc2Cl)C1 N1(C(C(C)C(C)O)=O)CCN(C(c2ccc(C(F)F)cc2F)=O)C(C(F)F)C1 Cc1nc2cc(C(=O)NCC3CC(F)(CNC(=O)C(C)CN(C)C)C3)ccc2s1 c1(CC)nc(C)c(C(=O)NCC2(NC(=O)C(CC)N(C)C)CCCC2)s1 c1(C(=O)NCC(C)CN(C)C(C2(CCN(C)C)CC2)=O)ccc(Cl)s1 c1(OC)ccnc2c1CCCC2NC(=O)NCCN1CCOC(C)C1 Cc1cc(O)ncc1C(=O)NC1CC=CCC1C(N1CCCC1CN(C)C)=O C(=O)(CC(C(F)F)C(C)(C)C)N(CC(C)(C)NC(C(C(C)C)(C)C)=O)C c1(OC(C)C(=O)NC2CCC2NC(c2cc(C(N)=O)c[nH]2)=O)cc(Cl)cc(Cl)c1 CC(C)(C)C(=O)Nn1cc(C(=O)NOCCN2CCCOC2)nn1 C1(NC(C(OC)OC)=O)CCCC(CNC(c2cn(C(C)(C)C)nn2)=O)C1 c1(C(=O)NCC(C)NC(C2(CC)CCCC2)=O)ccc(-c2cscn2)cc1 N#Cc1cc(S(=O)(=O)N(C2CNC2)Cc2ccc(-c3ccccc3)s2)ccc1F Cc1cc(NC(C2CCOCCN2C(C2CCN(C)CC2)=O)=O)ccc1Cl c1(C(=O)NCCCC(C)NC(C2CCCN2N=O)=O)noc2ncccc12 c1(CCC2(C(N(c3cccc(C(=C)C)c3)CC)=O)CCCC2)c[nH]c(=N)nc1C C1(C(=O)NC2(C(N3CC(C(CC)C)C3)=O)CCCCC2)CC(=O)NC(=O)N1 C1(F)(CNC(CCNC(C)=O)=O)CC(CNC(c2csnc2Cl)=O)C1 Cc1noc(C)c1C(C)C(=O)NCC(C)CN(C)C(C1CC(F)C1)=O N1(C(c2cnc(C)o2)=O)CC(NC(=O)Cc2cc(O)nc(O)n2)CC2(CC2)C1 Cc1cccc(F)c1C(=O)NCC1(F)CC(NC(c2ncc(C(F)F)s2)=O)C1 C1(O)(CC)CCN(C(C2CC(O)CN2C(c2cc(OC)n(C)n2)=O)=O)C1 C=CCCCC(C1CC1)NC(c1[nH]ccc1CNC(C1(SC)CC(C)(C)C1)=O)=O C1(C)(C(=O)NCCC(=C)CNC(C2(CC(C)C)CCNC2=O)=O)CNC(=O)C1 N1(C(C=CCC)=O)CCCCC1CCC1CCCN1C(c1cc(C)ns1)=O FC(F)(CCCn1cc(CCC2CCCN2)nn1)C(F)F N1(C(c2cnc(OC)nc2)=O)CCC2CCC(C1)N2C(=O)CC(C)(C)O O=C(C(CO)C(F)(F)F)NC(Cc1ccccc1Br)C(=O)N1CCC1CF C1(CNC(Cn2c(C)cnc2)=O)CCN(C(=O)C(C)N(C)C)CC1O c1(N2C(C)CNC(=O)C2)ncnc2[nH]c(=N)ccc12 c1(C(=O)NCCC2CCCN(C(CCC(C)O)=O)C2)cccc(C#N)c1 C(=O)(C(C)CC(C)(F)F)N(C1CCCN(C(=O)C=Cc2ccsc2)C1)CC C1(C)(C(N2CCCC(NC(c3cnc(CC)s3)=O)C2)=O)CCCC1(F)F N1(C(CCc2ncc(C)[nH]2)=O)C2CCC1CC(O)(CNC(=O)CCC1(C)CC1)C2 N1(C(Cn2c(C)c(Cl)cn2)=O)CCC2(CCC2)C(NC(C2CCCC(F)C2)=O)C1 N1(C(c2c(Br)ccc(C#N)c2)=O)CCC2(CC1)CC(NC(C1(CO)CC1)=O)C2 O=S(=O)(c1cc([N+](=O)[O-])ccc1Cl)NC1C(=O)OCC1CO C(=O)(C(O)CN1CCCC1)NCC1(CC(=O)NCC(C2CCOCC2)O)CC1 Cc1cn2c(n1)CCC(C(=O)NC1(CNC(C3CC4(CCC4O)C3)=O)CCC1)C2 C1(C(N(CCCNC(=O)Cc2ccc(F)nc2)CCC)=O)CCCCC1SCC C1(NC(=O)C(F)n2cccn2)CCCCCN1C(=O)COc1ccccc1 c1(C(N(CCNC(=O)C(C)Cc2ccccc2F)CC)=O)c(C)cccc1F Cc1ccc2c(=NC3CCCSC3)[nH]c(=NC(C)CCCN(C)C)[nH]c2c1 c1(C(N(CCN2CCN(C(c3ccc(C)o3)=O)CC2)C)=O)cc(F)c(F)cc1F CC12CC(C1)C(CN1CCCC(Sc3ccc(Cl)cc3)C1)CO2 N1(C(c2c(C)con2)=O)CCC(NC(c2cc(Cl)cc(C)c2N)=O)C(F)(F)CC1 c1(OCC)ccc(C)nc1C(=O)N(CCCOCCNC(=O)C=C(CC)CC)C CC(C)(CNC(=O)C(c1cccnc1)NC(=O)CCC1CCC(=O)C1)C(F)(F)F C1(C(=O)OC(c2ccc(Cl)cn2)C)CCC(C)(C)O1 Cc1cc(N)ccc1C(=O)NC1CCCCC1NC(C1CC1c1ccn(C)n1)=O c1(C(N2CC(COC)N(C(c3ccno3)=O)CC2)=O)c(Br)ccc2c1OCO2 c1(C(C)=O)cccc(C(=O)NCCOC2(C)CN(C(=O)CNC3CC3C)C2)c1 N#Cc1ccc(=NCC2(F)CCN(C(C3CCOC3)=O)CC2)[nH]c1 c1(C(N2CCN(Cc3ccc(F)cc3O)C3CC23)=O)ccc2cccnc2c1O N1(C(C(c2cccc(Br)c2)C)=O)CCCC(C)(CNC(=O)C(C)(C)F)C1 N1(C(C(C)C#N)=O)CCC(CNC(c2ccc3nc[nH]c3n2)=O)C(C2CC2)C1 Cc1cc(C)c(C(C)S(=O)(=O)NCc2c(F)cncc2Cl)c(C)c1C N1(C(CC2(C)CCCO2)=O)CC2CCN(C(c3coc(Br)c3)=O)C2C1 c1(C(C)C)ccc(C(N2CC3CC3(CNC(=O)CCOC3CCOC3)C2)=O)nc1 c1(C(N2C(CCNC(C3(CC)CC3)=O)C(C)CCC2)=O)cc([N+](=O)[O-])cc(C)n1 C1(NC(CNC(CC(C)C)=O)=O)CCN(C(c2ccc(CN(C)C)[nH]2)=O)C12CC2 C1(CCC)CN(C(c2cccnc2)=O)CCN1C(=O)NC1CCC(C)CC1 c1(N2CC3CN(Cc4nc(C)cc(OC)n4)C3C2)ccc(O)c(F)c1F c1(C2(C)CC2)cc(C(=O)NCCC2CSCCN2C(=O)C(C)(F)F)n(C)n1 N1(C(C2(C=C)CC2)=O)CCC(NC(=O)Cc2cc(F)cc(Cl)c2)C(O)C1 N1(C(c2c(NC(CN3CCC(C)CC3)=O)cco2)=O)CC(C)OCC1C c1(OC)ncnc(C(N2C(C(C)C)CCC2c2ccccc2)=O)c1F c1(CC)cc(C(N2CC=CC(NC(c3cc(O)nc(OC)n3)=O)C2)=O)cc(F)c1 c1(CC)ncccc1C(N1CCCC1C(C)(C)C(=O)N1CCC1CC1CCCC1)=O c1(NCCC(CC)OC)cc(=NC(C)C(C)CC)[nH]c(C(C)C)n1 C(CC(=O)N1CCCOC(C)C1)(C(F)(F)F)NC(C1(CSC)CC1)=O N#Cc1cccc(C(N2CCCC2CCNC(c2cnn(C(F)(F)F)c2)=O)=O)c1 c1(OC(C2N(CC(=O)NC(=O)OCC)CCC2)=O)cccc2cncn12 C1(NC(=O)Cc2ccns2)CC2(CCCCN2C(c2nnc(C(F)(F)F)s2)=O)C1 c1(C(N2CC(NC(Cc3ccc(C)cc3Cl)=O)C(F)C2)=O)ccc(C#N)c(F)c1F Cc1cc(C(=O)NC2CCN(C(=O)CCC3CCOC3)C2C2CC2)cc(C)n1 CC(C)CC(CNC(=O)CCc1cccc(O)c1)NC(=O)CCCC1CC1 c1(C(=O)NCC2(OCC)CN(C)C2)cnc(C)cc1C C(=O)(C(O)C(C)C)NCC(CCOC)NC(=O)CCc1nc(-c2ccsc2)no1 c1(C(=O)NCCCNC(CC(C)n2ccnc2)=O)cc(=O)cc[nH]1 C(C(CNC(c1cc(C2CC2)[nH]n1)=O)CO)NC(=O)Cn1cnnn1 c1(C(N2CC(CCCCC)C2)=O)c[nH]nc1CCNC(=O)C(C)(C)OCC c1(C(=O)NC2CC(C(=O)NCC3C(OCC)CC3)C2(C)C)cccc(O)c1F CCC(C#N)C(=O)N1CC(C)(NC(C2(CC(=O)OC(C)(C)C)CCOCC2)=O)C1 c1(C(N2CC3(CN(C(C4CC(=O)NC4)=O)C3)C2)=O)cnc2ncnc(O)c2c1 c1(CC(=O)NC2CC(OC)CN(C(=O)CCF)C2)ccc2c(c1)OC(F)(F)O2 c1(CC(=O)N(CC(C)CNC(c2c(Cl)cnn2C)=O)C)c(F)cccc1C#N N1(C(C(C(C)C)OC)=O)CCN(C(c2ccc(OC(C)C)nc2)=O)CC(C)(C)C1 C1(C(N(CC(C(F)(F)F)SC)CC)=O)CCC(=O)CC1C Nc1cccc2cc(S(=O)(=O)NC3CCCC3)ccc12 Cn1c(C(N2CC3CN(C(=O)CCCC4CCC4)CC3C2)=O)cc2ccccc12 N1(C(C(C)(C)N(CCC)CCC)=O)CCC(O)(CN(C)Cc2ccc(F)o2)CC1 C(=O)(C(=O)N=S(C)(C)=O)N1CC(C)C(NC(=O)Cc2cn3ccsc3n2)C1 c1(OCC)nn(C)cc1NC(=O)C#CCNC(C1CCC(C)C1)=O CCC(C(=O)NC(CNC(C1(F)CC1)=O)CC(F)(F)F)C(C)(F)F Cc1oc(C(=O)N(CCNC(C2CC2(C)Br)=O)CCOC)cc1CO Cc1nc(O)[nH]c1C(=O)NCC(Cc1ccccc1)NC(C1(F)CCCOC1)=O N1(C(C2N(C(CCCC)=O)CC3CC32)=O)CCC(O)CC(C)(C)C1 C1(NC(CC(CC)OC)=O)CC2CCC(C1F)N2C(=O)CCNC(N)=O N1(C(C2(OC(C)C)CCC2)=O)Cc2ccc(CN(C)C(C3CC3(F)Cl)=O)cc2C1 c1(C(N(CC(C)O)CCNC(c2c(C)nn(C)c2F)=O)=O)ccn2nccc2c1 C(=O)(C1CCCc2cccnc21)NCC(C(C)C)NC(=O)CCN(S(C)(=O)=O)C CCC(C)C(O)C(C)C(=O)N1CCCC(CC)C1C(N1CC(NC(=O)N(C)C)C1)=O c1(NCc2nc(CC)sc2)nc(N2CC(OC)C3(CC3)C2)nc2c1ncn2CC C(=O)(C1OC(=O)c2ccccc21)N(C)CC1CCN(C(C2C(C)C2)=O)CC1 N1(C(c2ccc(C(C)(C)C)[nH]2)=O)CCN(C(=O)CCCN=[N+]=[N-])C2COCC12 c1(C(N(CC(CNC(C2C(C)=C2)=O)(C)C)C)=O)cc(C)c(Cl)c(C)c1 c1(C(=O)NC2C(CNC(c3c(C)cc(OC)o3)=O)C2)cnc(O)c(C(F)(F)F)c1 N1(CC(=O)NC2C(NC(c3cc(O)ncn3)=O)COC2)CCOCC1=O N1(C(C(C)(C)O)=O)CCCC2(CC(NC(c3nccc(Cl)c3F)=O)CO2)C1 N1(C(CCC(C)OC)=O)CCCCC(NC(c2c(C(F)(F)F)coc2C)=O)C1 CCCC(C)(C)CC(=O)NC1CCN(C(c2cnc(C(F)F)c(C)c2)=O)C(C)C1 N1(C(C2N=C(C)SC2)=O)CC2(CCCC2NC(=O)CCOc2ccccc2C)C1 c1(NC(c2n(CC=C)nnn2)c2ccc(COC)s2)cccc2c1OCC2 N1(C(C=Cc2c(C)ncs2)=O)CCN(C(=O)COc2ccsn2)CC1CC1CC1 N#Cc1ccccc1CCC(=O)NCC1(O)CCCN(C(=O)COCC(F)F)C1 CC(C)(CNC1CCC(NC(=O)OC(C)(C)C)C1)C1=CCOCC1 N1(C(c2cnc(CC(C)C)[nH]2)=O)CCC2CCN(C(=O)Cc3cncnc3)C2C1 CCC(CC(=O)NC1CC(C(=O)NC(CO)CC(F)(F)F)C1)C(F)F C(=O)(C(C)(O)C(F)(F)F)NCC1C(NC(c2cn(C(C)C)nn2)=O)C1 N1(C(c2cn(CC(F)F)cn2)=O)CCCC(C)(C)C1C(F)(F)F CCC(C)C(O)C(=O)N(CCCN(C(=O)CC1CC2CCC1CC2)C)C CCC(C)(O)C(=O)NCCC(C)(C)NC(c1ccc(C)o1)=O N1(C(C=C(CCC)CCC)=O)C2CCC1CN(C(C1CC13CCC3)=O)C2 C(=O)(C1=CCC(F)(F)CC1)N(CC)CC.C1(=O)CCC(=O)NCC(C)N1 n1(C(C)C)cncc1C(=O)NC1CC(N(C)C(C2CC2C(F)(F)F)=O)C1 C1(N(C)C(c2cnn(C)c2)=O)CCN(C(C23CCCC2CC3)=O)CC1 Cc1cc(=NC2CCC(S(C)(=O)=O)C2)[nH]c(=NCCc2c(F)cccc2Cl)[nH]1 Cc1ocnc1CC(=O)N(C)CCN(C)C(C1(c2cncnc2)CCCC1)=O C1(NC(CCOCCN(C(C(C)OCCOCC)=O)C)=O)C(CO)C1(F)F c1(C(=O)OC)ccc(NC(C2CN(C(c3cccc(Br)c3Br)=O)C2)=O)c(OC)c1 C#CCCC(=O)NC(C)CNC(c1nnn(-c2ccccc2)n1)=O c1(C(N2CC(NC(C3(CC#C)CC3)=O)CC2(C)C)=O)cc(O)cc(F)c1F C12(C(=O)OC)CCCC1(C(N1CC(C)(NC(=O)CC3CC3(Cl)Cl)C1)=O)C2 C1(NC(CC(CNC(c2nocc2C)=O)OC)=O)CCc2c[nH]nc2C1 c1(CC(=O)NCCN(C(c2cccc(OCCC)c2)=O)C)c(C)nc(O)nc1O C(CC(=O)N1CCC(CCCNC(=O)CC(C)C(C)(C)C)CC1)(C(F)(F)F)OC C1(C(N)=O)COCC1C(=O)NC1CC(O)C1CC(=O)NC1CCCN1CC1CC1 c1(C(N(C(CCNC(c2c(C)cncc2)=O)C)C)=O)ncc(N)cc1Cl c1(C(=O)NC(C)CCN(C(=O)C(C)(Cl)Cl)C)cc2ccsc2s1 c1(C(=O)NCC(CNC(c2[nH]nnc2C)=O)OC)ncc2c(F)cccn12 c1(C(=O)NC2CN(C(C=C(CCN(C)C)Cl)=O)CC(O)C2)[nH]nc2ncccc12 C(=O)(C1=Cc2ccccc2OC1)N1CCC2(NC(C=COCC)=O)C(CC1)C2 C#CCCC(O)C(=O)N(C1CN(C(c2ncncc2Cl)=O)CC1O)C C=CCC(CNC(=O)CC1CN(C(C)=O)C1)C(=O)N1CCCCCC1 C1(COC)(NC(c2ncc(C(F)F)s2)=O)CCN(C(c2sc(C)cc2C)=O)C1 C1(CNC(CN(C(C(C)C)=O)C)=O)CC(O)CN1C(=O)CC(C)C1CCCO1 c1(C(N(CCC)CCNC(C2CSC2)=O)=O)cncc(C(C)(C)C)c1 c1(C(N2C(C(C)NC(c3c(C)cccn3)=O)CCC2)=O)nc2c(s1)CN(C)CC2 C(=O)(C(C)C(C)(F)F)NCC(C)CN(C)C(c1cc(I)c[nH]1)=O C1(c2n(CCC)nnn2)(NCc2ncc(CCC(N)=O)[nH]2)CCCCC1CC c1(C(C(=O)NCCCSC)N(C2(C#N)CC2)C)ccc(-n2ccnn2)cc1 c1(C(=O)OCC)c(NC(=O)C(C)CC)sc2c1CCC(C)C2 C1(NC(CC2CC(OCC)C2)=O)CN(C(C2C=CCS2)=O)CC1SC CC(C1=CCN(C)CC1)NC(=O)C(c1ccc(C#N)cc1)C C(=O)(C1=CCCC(C)(C)C1)N(CCCNC(c1ncccc1Cl)=O)C1CC1 c1(C(N2CC(CN(C)C(C3CC4CC3C4)=O)OCC2)=O)cnc2[nH]cncc1-2 c1(C(=O)NCC(=O)NC(C2CN(C(=O)CC(F)(F)F)CCO2)C)cc(Cl)cn1C Cc1ccc(C=CC(=O)NCCCCC2(NC(c3ccccc3C)=O)CC2)o1 N1(C(CCC2(C)CN(C(c3ccc([N+](=O)[O-])o3)=O)C2)=O)CC(O)C2(CCCC2)C1 C1(OCCNC(C(CC)OC)=O)CCN(C(c2cc(Cl)cs2)=O)CC1 N1(C(CN(C(C)=O)C)=O)CC(NC(c2cc[nH]c2C2CCCC2)=O)C(C2CC2)C1 CC1CN(C(c2cnc(C(C)(C)C)o2)=O)CC1NC(=O)CC1COCC1O C1(CNC(=O)Cc2ccco2)CN(C(c2cncc(C3CCCC3)c2)=O)C2CC12 c1(NC(c2ccco2)=O)ccc2c(c1)CN(C(C1(O)CCOCC1)=O)C2 N1(CCNC(c2[nH]cnc2-c2ccccc2)=O)CCOC(c2ccc(Br)cc2)C1 C(C)(C(=O)N=c1ccn(C(C)C)[nH]1)NC(C1CC(OCC)C1)=O N1(C(C)=O)CCOC(C(=O)NCCC(C)NC(C2CCC(C)O2)=O)C1 N1(C(c2cc(C)ns2)=O)CCC2C(CCN2C(c2[nH]cnc2C#N)=O)C1 C1(COC)CCN(C(=O)CC2CCN2C(C2(OC(C)=O)CCOC2)=O)C1 C(=O)(C(C(C)C)C(C)C)N1CC2C(CCNC(c3c(C)c[nH]c3)=O)(CC2)C1 N1(C(CN(CC#C)C(c2ccc(OC)s2)=O)=O)CC2CC(C)C2C1 C12(CNC(=O)CN3CC(OCC(F)F)C3)COCC(c3ccccc3)(C1)C2 C1(NC(C(C=CC)O)=O)CCC12CN(C(c1cnc(Cl)[nH]1)=O)C2 C1(C(N(C)CC2N(C(c3nc(C)n(C)n3)=O)CCC2)=O)CC2CC(O)CC(C1)C2 C1(Nc2cccc(C(=O)NCC3CC3)c2)CCCCN(Cc2ccc(Br)nc2)C1 N1(C(c2ccc(CC)cc2OC)=O)CCN(C(=O)C(C)(O)C(C)(C)C)CCC1C Cc1ccc(OCC(=O)N(C2CN(C(C3(O)CCSC3)=O)C2)C)cc1 c1(NC(CCC=CC)=O)ccc(NC(c2cc(Cl)cnc2O)=O)cc1C c1(C(=O)NC2CCN(C(c3cc[nH]c3)=O)CC2O)ccc2cc(Cl)ccc2n1 c1(C(=O)NCC(CC=C)NC(C2(CO)CCCO2)=O)cc(S(C)(=O)=O)cs1 c1(CC2(NC(=O)CO)CN(C(=O)Cc3cccc(Cl)c3)C2)ccc(CO)cc1 C(=O)(CCCC(=O)NC1CCC(C)N(C(c2ccc(F)cc2)=O)C1)NCC C1(NC(C2CCC3CC23)=O)CCN(c2nnco2)C12CCCC2 N1(C(C2C(OC(C)=O)C2)=O)CC2CC1CN2C(=O)C(C)=C1CC1 CC1CCN(C(=O)N(C2CC2)CC2CC3CC2C3)C1c1ccccc1 C(=O)(CCCC(=O)NC(C)(C)CNC(=O)C(C)Cc1c(C)noc1C)OC N1(C(c2cncc(Br)c2)=O)CCCC2(CCN(S(=O)(=O)c3ccc(Br)cn3)C2)C1 c1(CC)cc(C(N2CCC(NC(=O)CCOC3CCCC3)C(O)C2)=O)c(C)nn1 C12(CC)CC(C(=O)NCC3(C)CCN(C(=O)C4=CCSC4)C3)(CO1)C2 N1(C(C2CC(F)C2)=O)CCC2(CCN(C(C3(C4(O)CCC4)CC3)=O)C2)C1 N1(C(CCCOC)=O)CCN(C(c2ccnnc2)=O)CC1c1ccncc1 c1(C(=O)NC2CCCC2NC(C2(F)CC3(CCC3)C2)=O)c(OC(F)F)cccc1Cl C1(C(=O)NC(COC)CNC(=O)Cc2ccccc2F)C2Cc3ccccc3C12 Cc1cc(C(=O)NC2CC(O)(CNC(c3cccc(OCCF)c3)=O)C2)cn1C c1(C(N(C2CCN(CCCCC=C)C2)CC)=O)ccc2cccnc2c1 CC12CC(C(=O)NCC3CCCN3C(C3(Sc4ccccc4)CC3)=O)(C1)C2 S(=O)(=O)(c1ccc(NCC(C)O)c(Cl)c1)N(CCOC)CC.C1CC(C)N1 N1(C(Cc2cc(C)[nH]n2)=O)CCC2(CC(NC(=O)Cn3nnc(C4CC4)n3)C2)C1 c1(C(=O)NC2(C(=O)NC(c3nc(C)on3)C)CCN(C)C2)ccc(F)c(O)c1 Cc1cc(N)c(F)c(C(=O)NCC(CNC(=O)CC2(C)CCC2)CO)c1F N1(C(C2C(C)=CCC=C2)=O)CC2(CCCC2NC(=O)C=Cc2ccsc2)C1 C1(C(N(C)CCNC(=O)Cc2cccnc2)=O)CC(C)(C)C1C(F)(F)F C(CC(F)(F)F)(C(=O)O)NC(c1ccc(-c2ccc(C(F)(F)F)cc2F)nc1)=O N#Cc1cncc(NC2CCCCN(C(C34CC5CC3C4C5O)=O)C2)n1 N1(C(C(C)N(CC)CC)=O)CCC(C2CC2)(NC(c2cc(C(F)F)n(C)n2)=O)C1 N1(C(CCc2onc(C)n2)=O)CC(CC(N2CCN(C(C)=O)CC2)=O)CC1(C)C C(=O)(CS(=O)(=O)c1ccccc1Cl)N1C(C)CCN(C(COCCC)=O)CC1 S(=O)(=O)(c1cc(Br)cc2c1OCC2)N1C(C)(C(N(C)C)=O)CC1 Oc1c(CNCc2cnc(-c3cnn(C)c3)nc2)cccc1Cl C12(C(N3CC(OC)C(C(=O)NCCC4COCC4O)C3)=O)CCCC1OCC2 c1(N(CCOC)C)cc(N2CCOC(c3ccccc3Cl)C2)nc(C)n1 C1(NC(C2(SC)CC2)=O)CCCCC1NC(c1cc(C(C)C)nn1C)=O Cc1[nH]nc2ncc(N(c3ccccn3)C(C3CC4(CCNCC4)C3)=O)cc12 CC1CCC(C(=O)NCCC2CC(NC(c3ccc(CSC(F)F)o3)=O)C2)O1 N1(C(CC(C)(C)n2cc(CN(CC)CC)nn2)=O)CCn2cc(C)nc2C1 c1(CN(C2CCC(SCC)CC2)Cc2cc(Br)cnc2OC)cc(Cl)ccc1O N1(C(Cn2c(C)ncc2)=O)CC(NC(=O)CSc2ccccc2)C(F)(F)C1 n1(CC)nnc(C(=O)NCCN(C2CCCCC2)C(=O)CC2CCC(=O)N2)c1C N1(C(c2c(C)n(C)nc2)=O)CCc2cccc(O)c21 Cc1nc(N2CCC(CC(=O)N(C)CC3(O)CCCCC3)C2)n(C)n1 Cc1nccc(N2CCC(OCc3nc(C4CC4)cs3)C2)n1 C1(NC(C(CC=CC)NC(C2CCC2C(C)(C)C)=O)=O)CN(C)C2(CCC2)C1 CC(CC1CCCC1)C(=O)N(C(C)CCNC(=O)CCNc1ccccc1)C n1(CCNC(C2CN(C(C3CC4C=CC3C4)=O)CCC2O)=O)ccc([N+](=O)[O-])n1 C#CC1(O)CC(C(N2CCSCC2CCNC(c2cnc(CC3CC3)s2)=O)=O)C1 CCC(CC(C)C)C(=O)NC(CCC1CCC1)C(=O)Nc1cnc2c(c1)CCC2 C1(NC(C(CSC)NC(CC=CCCCCC)=O)=O)CCc2n[nH]cc2C1 N1(C(C(CC=C)(C)N(C)C)=O)CCC2CCN(C(C3(C)CC=CC3)=O)CC2C1 C(C(N=c1cc(Cl)nc(C)[nH]1)C1CC1)NC(c1ccc(CNC(CC)=O)cc1)=O c1(OC)ccc(O)cc1C(=O)N(CCCNC(=O)CCC(C)C)C(C)C Cc1cc(C(=O)NCCCCNC(c2ccsc2Br)=O)ncc1CO N1(C(CN(CC)Cc2ccccc2)=O)CC2(CC(NC(=O)C(C)C3CC3)C2)C1 N1(C(c2c(C)oc(Cl)n2)=O)C(CC(N2CCC(O)CC2C)=O)C2CCCC12 C12(C(N3CCCC(CCNC(C4CC(=O)NCC4)=O)C3)=O)CC(C1)S(=O)(=O)C2 C(C(=O)NOCC1CC1)=CCN(C(CN(C)CC1CCC1)=O)C N1(C(C(C2CCC(=O)N2)C)=O)C2CCC1CN(C(C13CC(CC4CC4)(C1)C3)=O)C2 N1(C(c2cn(C(C)C)nc2)=O)CCC2(NC(=O)C(=O)NC(C)C)CCCC12 c1(NC(C2CC(C(=O)OC)C2)=O)ncccc1Sc1ccc(C(=O)O)[nH]1 c1(OC)cnc(CNC(=O)C(O)CCNC(=O)C(C)C#N)cn1 Cc1ccc(N)c(C(=O)NCC2CCCC(CNC(=O)C(O)CC(C)C)C2)c1 C1(C(=O)NCC(C)N(C(=O)COCC2CCC2)C)CC(O)C1 c1(SC)ccc(C2(CNC(c3ccnc(SC)c3)=O)CCOC2)cc1 C1(CNC(c2csc(C(F)F)n2)=O)CC2(CCC2)CN1C(C1(O)CCSCC1)=O c1(CC(=O)NCCCCC(C)NC(=O)C=Cc2cncs2)cccc(O)c1F c1(CC)ccc2c(c1)C(CC(=O)N1CC(F)CC1CNC(=O)CC(C)O)C(=O)N2 C12(NC(=O)Cn3cc(C4CC4)cn3)CN(C(=O)C=CC(F)(F)F)CC1CS(=O)(=O)C2 C1(OC)CN(C(=O)C2=NOC(C)C2)CCC1NC(c1sc(C)nc1C)=O C(=O)(CCCn1cc(C2CC=CC2)nn1)NC1(CC=C)CC1 Cn1cnc2ccc(C(=O)NC3(CO)CN(c4nnc(C5CC5)o4)C3)nc12 c1(C2(NC(c3cscc3Cl)=O)CC2)ccc(N2CCOCC2)c([N+](=O)[O-])c1 CCCCC(CNC(=O)COCCOC)NC(c1csc(Br)c1)=O CC1CCCC(C(=O)NCC(C)(F)CNC(=O)CN2CCCCC2=O)CC1 C1(C)(C(N2CCC(CN(C)Cc3nnc(-c4ccco4)o3)C2)=O)CC(C)(C)C1 Cc1cc(C(=O)Nc2cccc(CCCO)c2)c(C)n1Cc1ccncc1 c1(C(=O)NC2CC3(CCN(C(C4CC=CCC4)=O)C3)C2)n[nH]c2cccc(F)c12 c1(OCC)cccc2c1OCC(C(=O)NCCN(C(c1ccon1)=O)CCl)=C2.C c1(NC)ccc(C(=O)NC(C2CN(C(C3(C)CCCO3)=O)C2)C)cc1 N1(C(c2ccc3sncc3c2)=O)CCCCC2(CCN(c3ncc(Br)cn3)C2)C1 C(C)(C)(C(=O)N(C)CCO)OCCNC(C=CC)=O Cc1c(C(=O)NC(C)(CNC(=O)C(C)CC(F)F)C2CCC2)cccc1F C1(COC)CN(C(=O)Cc2ccccc2Cl)CCN1C(=O)CC(C)C1CC1 N1(C(=O)NCCC(CC)O)CCC(CCN2CCCS2(=O)=O)C1C C(=O)(C1=COc2ccccc2O1)N(CC(C)O)CCNC(=O)Cc1ccc(Cl)s1 C(=O)(C(O)CC(N)=O)C(=O)CC1(N)CCC1.CC1(OCCN)CCOCC1 C1(CCNC(C2C(OCC)C2)=O)CCCN(C(c2c(C)ccnc2C)=O)CC1 Cc1[nH]nc(CO)c1C(=O)NCC1C2CN(C(c3cnc(N(C)C)cn3)=O)CC12 c1(C(=O)Nc2scc(C(N(C)CCO)=O)n2)cccc2c1oc1ccccc21 c1(C(=O)NCC2(NC(CS(=O)(=O)NC)=O)CCCC2)nccn2nccc12 c1(C(=O)NC2CCCN(C(c3ccn(C(F)F)n3)=O)C2)cc(Cl)ncc1F C#Cc1cccc(CC(=O)NCCOC(C)(C)CNC(C2SCCC2C)=O)c1 C1(CNC(C=CC=CC)=O)CN(C(c2ccncc2C)=O)CCC12CCOC2 C1(NC(=O)CC2C=CCC2)CCCN(C(c2cscc2C(F)F)=O)C1 c1(N(C)CCC2CC2)nc2cc[nH]c2c(=NC2CCC(=O)N(CCO)C2)[nH]1 c1(C(N2C(C(=O)NC(c3ccc[nH]3)=O)CCC2)=O)ccccc1NCC1CC1 CC(CN1CCOCC1)C(=O)NC1CC(NC(=O)C(C)c2cc[nH]n2)C1 N1(C(C(C)(C)NC(CCc2n(C)ncn2)=O)=O)CC2CC3CC2C1C3 O=CCS(=O)(=O)CC(F)(F)F.C1(COC)COCCN1C(=O)C(F)CC1CCCC1 N1(C(CCC(=O)NC)=O)CCN(C(=O)C(C)OCC(F)(F)F)CC1C(C)C c1(C(=O)NCC2(C)N(C(=O)CS(C)(=O)=O)CC(OC)C2)ccc2n[nH]cc2c1C n1(CC)ncc2cc(C(=O)NCC3CC(CNC(C4(Cl)CC4)=O)CO3)cnc12 Cc1cc(O)c(C(=O)NC2CCCC2NC(=O)C(C(C)C)N(C)C)cc1F C1(C)CCS(=O)(=O)CC1.C1(COC(C2C(OC(C)(C)C)C2)=O)CCCCN(C=O)C1 C1(NC(CCCCC=CC)=O)CCN(C(=O)COc2cccc(O)c2)CC1(C)C c1(C(=O)NCC(C)CN(C)C(c2cc(O)nc(O)n2)=O)ccnc2ccncc12 c1(C(=O)NC2C(NC(C(C)C)=O)CCC2)cccc(-c2cc(O)ns2)c1 C1(O)(C(=O)OCC)CCN(C(=O)CCC2CC2)CC1.c1(CCC)nc[nH]n1 c1(OC)cnc(Cl)[nH]c1=NC1CCCCC1NC(C12CCCN(CCC1)C2)=O Cc1cc(C(=O)NCC23CC(NC(=O)CC(F)(F)F)(CO2)C3)cnc1C(F)F c1(C(=O)NC2CCN(C(C3C(OC)C3)=O)C2)cc(O)nc(Br)c1 C1(CNC(C(C)SCC)=O)CC2(CO1)CN(C(C1(C)CS(=O)(=O)C1)=O)C2 Cc1scnc1C(N1CC(OCCN(C(C2(n3ccnn3)CC2)=O)C2CC2)C1)=O N1(C(CCN(C)CCO)=O)CCCCC1C(=O)NC1CC2CC2C1 C12(CCNC(C(C)(C)SC)=O)CCC1CN(C(=O)C(C)(C)n1ccnn1)C2 CN1CCOCC1C(=O)NCC1CCC(CNC(=O)CC2(C)CC(F)(F)C2)CC1 C1(CCC(=O)OC)(CN(C2CC2)Cc2nccs2)CC1(F)F c1(C(N(C(C)CN(C(=O)C(CCO)N(C)C)C)C)=O)cc2cc[nH]c2cn1 CCC(C(=O)NC(CC(C)C)C(=O)N1CC(C(=O)N(C)CC)C1)C(C)C c1(-c2n(C)ccn2)ccc(NCC2CC2C2CCC2)nc1 c1(CN2C(C(=O)NCC3CCC(=O)NC3)CC3(CC3)C2)c(Cl)[nH]c2ccccc12 N(C1c2ccccc2CC1NC(=O)Cc1ccsc1)C(C(CC)C(C)(F)F)=O N1(C(c2c(OC)scc2)=O)CCC2(CCCC2NC(=O)CCC(C)=O)CC1 C1(NC(C2CC=C(C)CC2)=O)CC2CCC(C1)N2C(C1(C)CC(C(F)(F)F)C1)=O c1(C(C)C)n[nH]cc1C(=O)NCC(C)(C)NC(=O)Cc1csc(Cl)n1 C1(F)(C(=O)NCC2(O)CN(C(c3c(C(C)C)ocn3)=O)C2)CCOCC1 Cc1c(C(N2CCCC(N(C)C(C3CCCCN3C)=O)C2)=O)[nH]c2ccccc12 Cc1ncc2c(n1)CC1CCC2NC(=O)C(=O)N(C)CC1CCCNC N1(C(C2C(COC)CC2)=O)CCN(C(C2(NC(=O)N(C)C)CC2)=O)CC1 c1(C(N(CCOC)CCNC(=O)CC2(C)CCOC2)=O)cccc2ccn(C)c12 C1(N(N2CCCCOC2=O)C(C)=O)C2CCCOC2C1(C)C.c12cccc(c1)S2 C1(CC=C)(C(=O)NCC2CC(C(=O)NCC(C)OCCO)CO2)CC=CC1 N1(C(Cc2c(C)nccc2)=O)CC(NC(=O)CC2(N3CCCC3)CC2)CC(O)C1 S(=O)(=O)(c1ccccc1C#N)Nc1ccc(CCNCC2(C(=O)OC)CC2)cc1 CC(C)C(F)(CNC(=O)CC1CCOC1=O)C(=O)Nc1cccc(CCO)c1 c1(OC)ccnc(C(=O)N(C(C)CNC(c2cnc(C(C)O)s2)=O)C)c1OC C(c1ccncn1)=CC(=O)NC1CC(CC(=O)NCC2(CO)CCOC2)C1 CC1Cc2cc(C(=O)N(C3CN(C(=O)CC45CCC(CC4)OC5)C3)C)ccc2O1 c1(CN2C(C(=O)NC3(C(=O)OC)CCC3)C3C(C2)C3(C)C)ccc(C)c(F)c1F C1(C2CCN(C(=O)C(CO)C(C)C)CC2)(CNC(C2(C#C)CC2)=O)CCOCC1 Cc1cccc(C(=O)NC2COCC2NC(c2ccc(CO)o2)=O)n1 C(C)(C)(CCC(=O)N1CCCC(O)(CN(C(=O)C2=C(C)CC2)C)C1)OC N(C(=NCc1cn(C)cn1)N1CC=C(c2c(F)cccc2F)CC1)C(C=C)C c1(C(C(=O)NC2CCCC(NC(c3nnn(C)n3)=O)C2)(F)F)cc(Cl)ccc1Cl c1(CC)ncccc1C(=O)NC(C)CCC(=O)NCCNC(C)=O C(=O)(C1=CC2(CCOCC2)C1)N1CCN(C(CCc2cc(C)on2)=O)C(C)C1 c1(CC)ccc(N(C(c2n[nH]c(C)n2)C(=O)NCCCF)CC)cc1 c1(C(N(CC(=O)O)Cc2scc(C)n2)=O)cccc2cc(Cl)ccc12 N1(C(=O)CCc2c(Cl)cccc2Cl)CC2CCC(N=c3[nH]nc(C(F)F)o3)CC2C1 Cc1cc(F)ccc1NC(C1C2CC1N(C(=O)COc1nc(O)nc(O)n1)C2)=O C1(C(=O)NOCC(C)(C)O)(NC(Cn2ncc(C)c2)=O)CCCOC1 C12CCN(C1CCOC)C(=O)N2.C=C(I)CC(=O)OC(C)(C)C N1(C(C2(C)CCC2)=O)CCC(F)(CNC(=O)CC23CCCC2C3)C1 c1(N2CCC(CC)C2)nc(NCC2CCCC2O)cc(C)n1 C(C(C)(C)C(C)O)NC(C(C)(C1CCC1)NC(c1cc(CC)[nH]n1)=O)=O CC1CCCC(C(N2CC(CCNC(c3cnnn3C)=O)C2)=O)CC1 C1(CCC)CCCC1C(=O)N(CCC(=O)NCc1ncc(C)o1)CC c1(CC(N2CC(C)C(NC(C3CCC(C(F)(F)F)C3)=O)C2)=O)ccc(O)c(F)c1 C(N=c1[nH]c2c(c(=NCc3cnc4ccccn34)[nH]1)CCC2)c1cc(CC)no1 Cc1cc(C)c(CC(=O)NC(C)C(C)NC(C2COCCOC2)=O)c(C)c1 c1(C(=O)NCC#CCNC(C(C)C2CCOC2)=O)cc2n(c1)CCCC2 c1(CNC(c2n(C(CC)C)nnn2)c2cn(C)cn2)ncc2c(n1)CCOC2 C1(C(=O)NCC(=C)CCNC(C2CCCS2(=O)=O)=O)CCOCC12CCCC2 c1(NC(N)=O)ccc(C(=O)NCC2(NC(C34CSCC3C4)=O)CC2)cc1 C1(NC(CNC(CCOC)=O)=O)CC(NC(=O)C=CC2CC2)C(O)C1 N1(C(C(C)N2C(=O)c3nc(OC)cc(n3)N2)=O)CCC2(CCCN(C)C2)C1.CC=CC C1(CNC(C2(COC)CC=CC2)=O)CN(C(C2C=CCCC2)=O)CCCO1 c1(C(=O)NC(CNC(c2n(CC)nnc2)=O)CO)cnn(CCO)c1C(C)C O=C1OC2CC(C(=O)NC3CCC(NC(C4(CCF)CCC4)=O)C3)CC2O1 Cc1cc(C(=O)NC(C)(C)CCC(=O)NCC(C)(C)CCO)c[nH]c1=N C1(F)(C(N(OC)Cc2ccccc2)=O)CCCN(C(c2cnc(C)cc2C)=O)C1 C=CCCC(O)CNC(C1(F)CCN(C(=O)CCNC(=O)COC)C1)=O C(=O)(C(C)CC(C)CC(C)C)NC1CCN(C(COCC#C)=O)C(C)C1 C#CC1(F)CCN(C(C2CC(C)CN(C(c3nc(C)ccc3F)=O)C2)=O)CC1 c1(C(=O)NC(CC)CN2CCCC2)conc1C(C)NC(=O)C=CC1CCC1 N1(C(CN(C)CC)=O)CCCC(C)(C)C1CNC(=O)C(C)Cn1cccn1 C1(C(=O)NCCN(C(c2ccc(C(C)=O)[nH]2)=O)C)CCC2(CC1)CC2 C(=O)(C1=C(C)CCOC1)NCC(C1N(C(CC2C(CC)C2)=O)CCC1)(C)C CCC(C)C(CNC(=O)CCN(C(=O)Cc1cn(C)cn1)C1CC1)OC C1(C(N(C2CCN(C(c3cnc(C)s3)=O)C2)C)=O)CCC(=O)N1CCC(F)(F)F N1(C(C(C=C)O)=O)CCN(C(c2cccc(CO)c2)=O)CC1CCC Cc1[nH]nc(C(=O)NC2CC2NC(C2(N3CCCCC3=O)CC2)=O)c1Cl c1(C(=O)NCC(C)(C)F)cc2cc(-c3cccc4c3OCCO4)cnc2[nH]1 c1(C(=O)NC2(CC(=O)NC(C(N)=O)C3CCCC3)CC2)cccnc1 C1(O)(CNC(=O)CC2CCCCO2)CCN(C(=O)C(c2ccc(Cl)nc2)(F)F)C1 C1(NC(C2N(C(CCNC(COC)=O)=O)CC3(CC3)C2)=O)CC2CC1OC(=O)N2 c1(C(=O)NC2(CNC(C3C(OCC)C3)=O)CCCC2)cccn2nnnc12 CCCS(=O)(=O)CC(=O)NCC(CO)NC(=O)CC1CC=CCC1 c1(C(C(=O)NC2(C)CC2)N(c2cn(CC)nc2)CC)ccc2c(c1)CCCO2 Cc1cccc(NC(=O)C(n2cc(CCCO)nn2)C)c1S(C)(=O)=O C(=O)(CC(CC)CC)NCC(=C)CCNC(=O)CCc1cccc(OC)n1 CC1OC2(C)CC1(C(N1CCC1CNC(C1CC(F)C1)=O)=O)C2 C1(C(=O)NC2CC(NC(C(c3cnn(C)c3)C)=O)C2)C2COCC12 N1(S(c2c(C)onc2)(=O)=O)CCCC2(CCN(C(=O)CC(C)(O)CC(=O)O)C2)C1 c1(OCCC(=O)OC(c2ccc(C)cn2)CN(C)C)cc(Cl)ccc1Cl CN1CCCC(C(N2CCN(C3CN(C(=O)CC4CCSC4)C3)CC2)=O)C1 C1(CC)C(C(=O)N(CCC(N)=O)CC)CCN1C(C1CCN(C)CC1)=O c1(C(=O)NCC2(O)CC(CNC(=O)Cn3ccnn3)C2)ccc(Cl)cc1 N1(C(c2n(CC)ccn2)=O)CC2CC1(CNC(=O)C(C)(C)OC)C2 C(C(C(=O)N(CC(O)CC)C1CC1)C(C)(C)C)NC(COCC)=O C1(C(=O)NC2CCC2O)(CC)CN(C(c2c[nH]cc2CC)=O)C1 CCCCCCCCC(=O)N1CCC2CN(C(c3scc(OC)c3OC)=O)CC12 N1(C(c2cccc(OC)c2F)=O)CC2CCC(C1)N2Cc1cn(C(C)(C)C)nn1 c1(OC)nc(C(=O)NC(C)(C)CNC(c2cn(C3COC3)nn2)=O)ncc1F c1(C(N2CCC(C(C)(C)NC(C(COC)C)=O)C2)=O)cc2occc2s1 C1(NC(C(CC)OCC)=O)CCCCN(C(=O)CNC(=O)OC(C)(C)C)CC1 C(=O)(C1=NNC(=O)CC1)NC(CCNC(c1cc(C)n(-c2ccccc2)n1)=O)C c1(C(N2C3C(NC(C4C5CC6C(C5)C46)=O)CC(C3)C2)=O)cc2c(s1)CCOC2 C(CC=O)N(CC)CC.C(CCOCC(=O)N)OCCN(CCC)CCC C(CCCCCn1cc(-c2nnccc2C)nn1)N(C(CCOC)=O)CC(F)(F)F Cn1ccc(C(C)(C)C(=O)NC2CN(C(=O)CC3CC3c3ccccc3)C2)n1 c1(C(=O)NCCN(C(c2ccc(O)nc2C)=O)CC)ccc(C)cc1[N+](=O)[O-] N1(C(C(CC=C)C)=O)CC2(CCCN(C(=O)Cn3cnnc3)C2)C1 N1(C(Cn2nc(C)n(C)c2=O)=O)CCCC2(NC(c3cn(C)nn3)=O)CC2C1 Cc1nc(-c2nn[nH]n2)ccc1NC(C1CCCN(c2nccs2)C1)=O Cc1cncc(C(=O)NC2CCN(C(c3cc[nH]c3C3CC3)=O)C2C(C)C)c1C C1(CNC(c2nnn(CC)c2C)=O)C(C)CCCN1C(c1cc(=O)cc(Cl)[nH]1)=O N1(C(c2c(C)oc(Cl)n2)=O)CC(NC(=O)C(C)(C)C2CC2)CC12CCOC2 c1(C(N2C(C(C)(C)O)CCC2)=O)ccc(F)nc1 c1(C(N2CC(C)(CCC(=O)N3CCC3CC3CCCC3)C2)=O)ccc(F)cn1 c1(N(CC(=C)C)C)nc(=NCC23CCCCC2C3(F)F)[nH]c2c1CSC2 c1(C(=O)NCC2(C)CC(NC(c3ccoc3CC(N)=O)=O)C2)ccc(F)cc1F c1(CNCC2OC(C)=C(C(=O)OC)C2)nc2ccc(Cl)cc2n1C C1(OC)(OC)CC(Oc2ccccc2C#N)C1(C)C.C1CC(=O)O1 C1(C(=O)NCC2CC3(CCC3)CN2C(=O)Cn2nccn2)CCc2nn[nH]c2C1 Cc1cc(C(=O)NC(c2cnn(CC3CCC3)c2)C)n(C(F)F)n1 CCCC(C)(C)CC(=O)NC1CCCCN(C(c2snnc2C2CC2)=O)C1 C(CCCC(=O)N(CCN(C(=O)CS)C)C)NCCS.C(=O)C(F)(F)F.C1CN1 N1(C(C(CC)N2CCCC2=O)=O)CC(OC)CC1CNC(=O)CC(C)C1CC1 c1(C(=O)NC2CCC(NC(c3cc(COC)[nH]n3)=O)C2)ccc2[nH]c(=N)oc2c1 c1(OCC(=O)NCC2OCCC2C(N2CCCC2C)=O)ccccc1.C(N)(=O)N C(c1ccc2[nH]ccc2c1)=CC(=O)NCC(C(C)(C)O)F C1(NC(c2ccnnc2O)=O)CN(C(c2ncccn2)=O)CC1F Cc1ccc(-c2nnc(C(C)NC3CC3c3ccc(Br)s3)o2)c(C)c1 C1(O)(CNC(c2cc(Br)ccc2O)=O)CCCN(C(=O)CC2CCCCO2)C1 CCCCCC(CCCCC)CC(=O)NCC1CC1NC(C1CN(C)C(=O)N1)=O C(=O)(C(C(=O)OOC(F)(F)F)OC)NCC1CN(C(CCSCCCOC)=O)C1 c1(OC)ccc(OC)c(C(=O)NC2CC(NC(=O)C=CC3(C)COC3)C2)n1 N1(C(C(CN(CC)CC)F)=O)CCC(COC)(NC(c2ccnn2CC)=O)C1 n1(CC(=O)NCC(C)N(C(=O)Cc2ccc(Cl)cc2Cl)C)cc(F)ccc1=O c1(NC(C2C3(CCN(Cc4nc(C)oc4)CC3)C2)=O)cc2c(cc1Br)OCCO2 C1(C(=O)NCc2cc(C#N)sc2)CCC2CCC1N2C(C1CC2CC(=O)C1C2)=O N1(C(c2nnn(C(C)(C)C)n2)=O)CC2=C(C1)CN(C(=O)C(C)n1cccn1)C2 C1(NC(c2n(C)ncc2)=O)CC2CC1CN(C(C1CCC1)=O)C2 c1(C(C(=O)NC2CN(C(C3(C)CCC3)=O)CC2O)O)ccc(F)cc1Br c1(C(=O)Nc2n(CC)ncc2)nc2ccc(-c3cc4ccccc4[nH]3)cc2s1 c1(C(=O)NC2(CC)CN(C(c3cnc(OC)c(C)c3)=O)C2)cc(C)c(C)nn1 c1(NC(C(CCF)NC(C(C(=O)OC)OC)=O)=O)cnc2ncnn2c1 c1(C(=O)NCC(C)(C)NC(=O)Cc2ccco2)ncc[nH]c1=O C(=O)(C(C)S(N)(=O)=O)N1CC(OCCC(=O)NC2C(C(=O)OC)C2)C1 Cc1cc(CC(N2CCC(C(C)NC(=O)COc3ccon3)C2)=O)cc(C)c1 c1(-n2cc(CSC)nn2)ccccc1CCC(=O)NCC(C)(N)Cn1cccn1 O=C(CC1OCCc2ccsc21)NC1(CNC(c2c[nH]nc2C(F)(F)F)=O)CC1 N1(C(C(=O)NCC)=O)CC(NC(c2cnc(OC)s2)=O)CC12CCCC2 c1(OC)nc(C(N2CCCC2CNC(=O)C2=CC(C)(C)C2)=O)cc(O)n1 N1(C(c2cc(C(C)=O)cn2C)=O)CCC(F)C(NC(=O)CN2CCC(O)CC2)C1 c1(C(=O)NCC2(F)CCN(C(C3CCCOC3)=O)C2)cc(F)cc([N+](=O)[O-])c1 N1(C(CCS(C)(=O)=O)=O)CCC2(C1)CN(C(C1CCC(N=[N+]=[N-])C1)=O)C2 N1(C(C(C=C)CC)=O)CCC(C)(C)C(CNC(=O)CC(C)(C)SC)C1 C(=O)(CC(CCC)NC(=O)C(c1ccn(C)n1)C)N(C1(C#C)CC1)C1CC1 C1(CNC(c2cc(C)c(C(F)F)cn2)=O)CC2CCC(C1)N2C(=O)C=CC1CC1 C1(NC(Cn2nnc(=N)[nH]2)=O)CC2CC(NC(C3CCC3)=O)C1C2 n1(CC)nccc1C(=O)N(CCC(C)NC(=O)C(O)CSC)C Cc1cnc(C(=O)NCC2(C)CCN(C(c3cscc3C3CC3)=O)C2)cc1C#N Cc1oc([N+](=O)[O-])cc1C(=O)NCC1CC(O)(CNC(C2CC23CC3)=O)C1 c1(C(N(CCN(C(c2c(C)nsc2)=O)C)C(C)C)=O)n[nH]c(C2CC2)c1C N1(C(CC2CC(=O)NC2)=O)CC(NC(C2CN(CC(F)(F)F)C2)=O)C2(CC2)C1 C(CCC(C(=O)NC(c1ccccc1)C)NC(c1c[nH]nc1Cl)=O)OC C1(CCC(N2CC(CCNC(C=NOC)=O)C2)=O)CCC(=O)NC1 CCC(C)CCCC(=O)NC1(CCC(=O)NCC(O)CC2CCC2)CCC1 c1(-n2c(C(=O)OC)cnn2)c(Cl)cccc1Cl.C1(C(=O)OC)CN2CC1C2=O c1(C(N2CC(O)(CCNC(C3CC(C)OC3)=O)C2)=O)cccc2c1CCS2(=O)=O Cc1onc(Br)c1C(=O)NC(C)CCCNC(c1ccccc1F)=O c1(CNC(CC(C)C)=O)ccc(C(=O)NCC2(CO)CCOC2)nc1 C1(CC#C)(C(=O)NC(CN(C)C)CC)CCN(C(c2sccc2Cl)=O)C1 C1(CC(=O)N(C(c2ccc(Cl)c(Cl)c2)C)C)CC2CNCC2(c2ccccc2)C1 C1(C(=O)Nc2c(C)nc(-c3ncc[nH]3)s2)COC2(CO)CC1C2 Cc1nc(C(N2CC(CNC(c3csc(CO)n3)=O)C(C)C2)=O)c2ccccn12 CCC(CC(C)CO)NC(=O)CCCCN(C(=O)CCC1(C)CC1)C Cc1ccc2c(c1)N(C(c1coc(CNC(=O)COCC3CCOC3)n1)=O)CC2 N1(C(c2ccc(CCCC)cc2)=O)CCCC2CN(C(=O)CCC(C)SC)CC12 C(C(CC)(CC)NC(=O)C(O)C(C)c1ccccc1)NC(C=C(CC)CC)=O CS(=O)(=O)c1ccc(F)c(NC(=O)Nc2cc3n(n2)CCNS3(=O)=O)c1 CC(C)(CC(=O)NC1CCC(CNC(=O)Cn2cnc([N+](=O)[O-])c2)C1)C(F)F N(C(=NCCCF)NCc1ccoc1)CC(C1CCC1)OCC c1(C(C)=O)cccc(C(=O)N(C)CCC2CCN(C(c3ccsn3)=O)CC2)c1 N1(C(c2c(C)n(C)cn2)=O)CCN(C(=O)CCCNS(C)(=O)=O)CC(O)C1 C(=O)(C(C)(C)C(=O)NCCCN(C(=O)COCc1ccccn1)C)OC C=CCC(C)(O)C(=O)NCC(O)C(=O)Nc1cnc(F)nc1 N1(C(Cn2ccc(C)cc2=O)=O)CCC2C(NC(C3(F)CCCCC3)=O)C2CC1 S(=O)(=O)(c1cnc(NC2CC2)c(Cl)c1)NCC(c1c(OC)cccc1)O C1(C(=O)NCC2CC(NC(CCC=C(C)C)=O)C2(C)C)SC2C=CC1CC2 Cn1cnnc1SCC(=O)NCC1(C)CC(NC(c2cc(Br)c[nH]2)=O)C1 c1(C(=O)NC(C(C)O)CO)cc(F)ncc1NCc1ccc(C(F)(F)F)c(F)c1 CCC(CC)C(=O)N1CCN(C2CCN(C(=O)C(O)C3CCC3)C2)CC1 C1(C(F)(F)F)CCC(NCCC2CC3CCC2O3)CN1 N1(C(C2(c3c(C)c[nH]n3)CC2)=O)CC(CNC(C2C(F)(F)C23CC3)=O)C(O)C1 N1(C(C2(C)CC3CC3C2)=O)CCC2(C1)CN(C(C1CCCCC13CC3)=O)C2 c1(C(=O)NC2(C(N(C)Cc3ncc(C)o3)=O)CCC2)cnccc1C C1(C(F)(F)F)(NC(C)=O)CCN(C(c2csc(I)c2)=O)CC1 C(=O)(CC(C)CC(C)C)N(CC(=O)NCCCCC#C)C1CC1 C(=O)(C#CC1(C)COC1)N1CCN(C(C2(CO)CCSCC2)=O)CC1CF.CCO Cc1cc(O)ccc1C(=O)NCC1CCC1NC(=O)C(C)(C)C1CCCCO1 N1(C(C2CC(C(F)(F)F)(OC)C2)=O)CCC(C)(NC(c2ccc(C)cc2)=O)C1 CC1(C)CC(CC(=O)NC2CCC2)N(C(C2CC(=O)CCO2)=O)C1 c1(CCNC(COCCNC(=O)CCSC2CC2)=O)cccc(O)n1 C1(C(=O)NCCN(C(CC)C)C)(NCCO)CCc2cc(Br)ccc2C1 c1(CC)ncc(Cl)c(C(=O)NC(C)CCCNC(c2sc(=N)[nH]c2C)=O)n1 c1(OC)ccc(CN2CCCC(C)(CSC)C2)cc1OC N1(C(CSC)=O)CC2CCOC2(CNC(c2n[nH]c3c2CCOC3)=O)C1 C(=O)(C=CS(C)(=O)=O)NCC1N(C(CCC(=C)Cl)=O)CCC1C N1(C(c2n(CCC)ncc2)=O)CCC2(CCN(C(=O)C(C)NC(N)=O)C2)C1 C(=O)(CCCCCn1cc(C(C)(C)N(C)C)nn1)NCCc1ccn(C)n1 C1(COC(COc2cccc(C(C)=O)c2)=O)CCc2nc(C)[nH]c2C1 c1(C(C(=O)N(C)OC(c2cn(CC)nn2)(CN)OCC)C)ccccc1Cl C1(C(=O)NCC(CNC(=O)CCc2cnn[nH]2)O)CCCSC1 c1(CC)ccnc(C(=O)NC2CCCC(C(=O)N(C)CCC3CC3)C2)c1 O=C(C#CC1CC1)NC(CNC(=O)Cc1ccccc1OC(F)F)C1CC1 c1(OC)ccc(CCC(=O)OCC2CCCN2C(C2C3CCOCC23)=O)cc1F O=C1CN(C(=O)CCCC2(NC(c3cccnc3)=O)CCC2)CCCN1 CC(C)CC(F)(F)C(=O)NCC1(C)CCCN1C(=O)C(N1CCOCC1=O)C c1(NC(C2CCN(C(=O)NC)C2)=O)ccc(NC(=O)Cc2ccsc2)nc1 c1(C(=O)NC(C)CCNC(=O)CSCc2ccncc2)[nH]cc2c1CCC2 C1(C(=O)OC)CCCN1S(=O)(=O)N(C1CC1C1CC1c1ccccc1)C(C)C CC1=C(C(=O)NCCC(C(C)C)NC(=O)CCC(C)c2ccccc2)SCCO1 CC1Cc2ccccc2C1Nc1nccc(=NCC2(C)CCOC2)[nH]1 C1(C(N(CCCN(C(C(=Cc2cccs2)C)=O)C)C)=O)CC(C)(C)OC1(C)C c1(CC)nnc(N(C)CC)n1CCC1CCCCO1 c1(C(=O)NCCCNC(CC(C)C2CCCO2)=O)cc(Cl)c(F)cc1Cl c1(C(N(C2CCCN(C(C(C)OCCC(C)C)=O)C2)C)=O)cc2occc2n1C c1(COCC)nc(N2CCCCC(CNC(C3C(C)OC(C)C3C)=O)C2)cc(C)n1 C=C(Cl)C(C)(C)C(=O)N1CCOC(CNC(=O)Cn2cc(C3CCOC3)cn2)C1 N1(C(C(=O)NCC2CC2)=O)CCCC1CN(C(C1(Cl)CC1(F)F)=O)C1CC1 C1(NC(c2cncc(-n3c(C)c(C(=O)O)cn3)c2)=O)CCS(=O)(=O)C(C)C1 C1(NC(C2C(C)(C)C(=O)NC2)=O)CC2(CCN(C(c3[nH]cc4c3CCC4)=O)C2)C1 N#CC12CC(C(=O)NCCC3CN(C(C4CC5CC5C4)=O)CCO3)(C1)C2 c1(CCC(=O)NC2C(NC(C(CN(C)C)O)=O)C2)ccc2ccccc2n1 C1(NC(C(c2scc(C)n2)C)=O)CCOCC1NC(c1cn(C)nn1)=O c1(CC)noc2ncc(C(N3CC(CNC(C4CCCC4C)=O)C(O)C3)=O)cc12 CC1C(NC(c2cccc(CC#N)c2)=O)CCN1C(=O)C(F)CC1CCOCC1 CC(C)CC(C(=O)NC)N(C(=O)CC1CCN(CC#N)C1)C Cc1ccc(C(=O)NC(CC2CC2)C(=O)NC2CC(CC(N)=O)C2)c(C)n1 N1(C(CCC(=C)C)=O)CC(NC(c2cnc(C)nc2C2CC2)=O)CCC(O)C1 c1(C(=O)NC(C(N2C(C)(CCC)CC2)=O)CO)ccncc1F C1(CC(=O)NCCCN(CC)Cc2ccc(NC(C)=O)cc2)CCCS1(=O)=O C(=O)(CC(C1CC1)NC(C1COCCO1)=O)N(C1CCOC1=O)C N1(C(c2c(C)onc2)=O)CCC(O)(CCNC(=O)Cc2ccsc2Cl)CC1 CC1CC2CN(C(C3C4CC(=O)CC34)=O)CC2N1C(C12COCC1C2)=O CC1(C)CC(NC(=O)CCC(=O)N2CCOCC2)CN1C(=O)C=C1CC1 C1(CNC(C(CCC)C#N)=O)CC2CCCC2N1C(=O)C(c1nc(C)cs1)C C=CCCC(F)(F)C(=O)N1CC(CNC(C2CCCCCC2)=O)C(F)(F)C1 N1(S(C(C)C)(=O)=O)CCC12CCN(C(=O)CSc1ccncc1)CC2 C1(NC(c2c(C)ocn2)=O)CCC12CN(C(=O)CCS(C)=O)C2 c1(C(N(CC(C)(C)NC(c2c(C)cno2)=O)C)=O)cc2scnc2[nH]1 c1(NC(C2N(C(c3c(C)ccc(C)c3)=O)CC(O)C2)=O)nc2ccc(Br)cc2o1 C(=O)(C(C)(C)CO)NCC(CCOC)NC(c1cnn(CCO)c1N)=O C12(CC(F)C1)C(=O)N2.CC(C(=O)NCCCCn1ccnc1)N1CCCC1 C1(NC(c2c(C(C)NC(=O)CCCCNC(N)=O)noc2)=O)C(=O)NCCC1C CC1CN(C(c2cc(C(F)F)ccn2)=O)CC1CNC(c1c[nH]nc1Cl)=O C1(C(=O)NCCCN(C)C(c2cc(C(F)F)nn2C)=O)CCn2c(O)nnc2C1 c1(CC)nc(N2CCC(C)(CN(C)C)C2)cc(NCCOC(C)(C)C)n1 N1(C(c2ccc(CC)s2)=O)CC(CNC(=O)Cc2csc(C)c2)CC1(C)C N1(C(C(CO)NC(N)=O)=O)CC(NC(c2cc(Cl)cnn2)=O)CC12CCCC2 CCS(=O)(=O)CC(=O)NC(C1(C(=O)NCCn2cccn2)CC1)C C1(N(C(=O)COCc2ccnn2C)C)CC2CC1N(C(C1(C#N)CC1)=O)C2 N1(C(CC2(C)CC2)=O)CCN(C(=O)COc2ccc(F)cc2)CC(O)C1 C1(C(N2CC3CC3C2)=O)Cc2nccnc2CN1C(C1CC1(F)F)=O Cc1cc(C(=O)NCC(C)CN(C(=O)C2=CC(O)CCC2)C)cc2nc[nH]c12 c1(C(=O)NCC2OCCN(C(Cc3cc(C)ncc3)=O)C2)cc(CO)ccc1C c1(C(=O)NC2CN(c3ncnc4c3CCC4)CC2F)c[nH]c2c(Br)cccc12 CC1(CNc2ncc(I)cn2)CCCN(C(c2nccnc2N)=O)C1 C(CC(=O)NCc1ncc(CO)[nH]1)(C(F)F)NC(C1CCC(C)(C)C1)=O C(C)(CC(=O)NCCOCCN(C(=O)CCc1nccs1)C)(C(F)F)N(C)C C1(NC(Cc2cnc(C)s2)=O)CCN(C(=O)CCN(C)CCO)C1C(C)(C)C CCC1=NOC(CC(N2CCN(CCNC(N3CCCC(CC)C3)=O)CC2)=O)C1 c1(OCC)ccsc1C(=O)N(CC(CC)NC(c1cnc(O)o1)=O)CC C1(F)(CNC(CNC(c2ccc(C)s2)=O)=O)CC(N=c2cc(C)c(C#N)c[nH]2)C1 C1(C(N2C(CNC(CC3COCC(C)(C)O3)=O)CCC2)=O)CCC2CCCCN12 C(C)(CCCC(=O)NC1CCCCC1C#N)NC(C1(C#C)CCCC1)=O n1(CC)cnc(C(=O)NC(C)C(C)NC(C2(c3ccsc3)CC2)=O)c1 C(C(CC(F)(F)F)C(=O)NCC1COCCOC1)NC(c1nccc(CC)c1)=O N1(C(C2CCN(OC)CC2)=O)CCCC2(CCCCC2NC(=O)C(C)N(C)C)C1 C(=O)(C1=CCCCC1C)N(CCNC(c1ccc(-n2ccccc2=O)cc1)=O)CC C1(OC)CN(C(=O)C(C)Oc2cccnc2)CC1NC(=O)CC(C1CC1)C1CC1 N1(C2C3C(CCCC2)C(=O)CN(CC#C)C3=O)CC(O)CC1C(N)=O N1(C(c2ccc(OC)cc2C)=O)CC2CCC(C1)N(C(c1cn(C)c(O)n1)=O)C2 C(CC(CC)C(=O)N1CC(NC(=O)CCc2c(C)noc2C)C(CO)C1)=CC N1(CCN(C)C)CCN(C(=O)CCOCCCNC(C2(C)CCC(=O)N2)=O)CC1 CCCC(C(=O)NCCNC(=O)C(C)CC)NC(c1ccccc1C(C)(F)F)=O N1(CC=CC(=O)NCCCN(C)C(C2CC(F)C2)=O)CCCC1 C=C(Cl)CC(C(=O)N1CCC1(C)CCC)NC(=O)CC1C=CCC1 C1(O)(CNC(CC2(N(C)C)CC2)=O)CCCN(C(C2CC2C(N)=O)=O)CC1 C1(C)(C(N2CC(C(C(=O)NCC(COC)C)O)C2)=O)CC(F)C1 c1(-c2nc(CSCc3nc(CC)c(C)o3)on2)ccc(C=CC(=O)O)cc1 CC(CC(=O)NC1CCCN(C(c2ccsc2C#N)=O)C1C)P(C)(C)=O C1(NC(c2cnc(C(F)(F)F)s2)=O)CN(C(=O)C=Cc2cn[nH]c2)CC2CC12 C1(C(=O)NC2(C)C(NC(C(Cc3c(C)nc[nH]3)O)=O)CCC2)CC2(C1)CC(O)C2 C1(C(N2CCCC(CCNC(C(CSC)(C)C)=O)C2)=O)CC(F)(F)CCC1(C)C c1(C(=O)NCCCN(C(Cc2ccc(C)cc2)=O)C)cnc(O)c2ncccc12 N1(C(CC(=O)NCC)=O)CC(=O)CC1C(=O)NCc1cccs1 Cn1ncc(C(=O)NC2CCCC(NC(c3csc(Br)c3)=O)C2)c1F c1(C(N2CC(CC=C)(NC(c3cncc(C)n3)=O)C2)=O)cn2c(n1)CC(C)CC2 C1(NC(C(C)(C)c2ccccc2)=O)(CO)CCN(C(c2ccccc2Cl)=O)C1 Cc1ccc(C2(C(=O)NC(C)CNC(C3CC3c3cncn3C)=O)CC2)c(F)c1 c1(C(N(C2CCN(c3ncns3)C2)C)=O)coc(Br)c1 C1(OC)COCCC1N1CCN(CC2CCCC2)CC1.C12CCCN1NC2=O C(=O)(C(F)C1=CCCCC1)NC1CCC(N(C(Cc2c(C)n(C)nc2)=O)C)CC1 N1(C(=O)NCC23CCC(F)(CC2)C3)CCc2ccc(F)cc2C1 C1(C)(C(=O)NC(C)CCCNC(c2ncn(C(C)(C)C)n2)=O)CCC(F)(F)CC1 N1(C(c2c(C)nn[nH]2)=O)CCC(C2CCN(C(=O)Cn3cncn3)CC2)C1 c1(C(=O)NC(C(C)NC(CN(C(C(C)C)=O)C)=O)C)cnc(N2CCOCC2)nc1 C(CN=c1[nH]cc(C#N)c(=N)[nH]1)n1c(=O)n2cnn(-c3ccc(F)cc3)c2c1 C(C)(C)(CC(C)N1CCC(C(=O)NC)CC1)C(N1CCCCC1)=O c1(C(c2nnnn2C2CCCCC2)NCCCC=C)cnc2n1CCC2 N1(C(C(CC(=C)C)C)=O)CCC(F)(F)C(CNC(=O)CN(C2CC2)CC)C1 c1(C(=O)NCC2C(NC(=O)Cn3ccccc3=O)COC2)ccc(Cl)c(Cl)c1O N1(C(CCNC(C(n2c(C)ccn2)C)=O)=O)CC2CC(O)CC2C1 N1(C(CC2(C)OCCO2)=O)C(C(=O)NCCN2CCNC2=O)CCC1C1CC1 C(=O)(C1=NN(C)C(=O)CC1)NC(COC)C(=O)NC1CC(OCC)C1.C(C)=O C12(NC(C(CC)C3CCOCC3)=O)CC(CNC(c3csc(C)c3)=O)(C1)OC2C C1(NC(CSCCN(CC)CC)=O)CCN(C(=O)CCn2c(C)csc2=O)C2CC12 C(CCC1CCC1)(C(=O)Nc1cncc(F)c1)NC(C(C)=O)=O O=C1Nc2ccc(NC(C3CCCCC(O)C3)=O)cc2C1=O C12(NC(C)=O)CCN(C(c3cn(-c4ccc(Cl)cc4C(F)(F)F)nn3)=O)CC1C2 Cc1nc(C(=O)N(CC(O)CNC(c2nc(Cl)c(Cl)s2)=O)C)ccc1[N+](=O)[O-] Cc1ccc(C(=O)NC(C(=O)NC2CCCCC2(C)C)C2CC2)cc1O C1(C(=O)NCc2scc(CNC(Cn3ncn(C)c3=O)=O)n2)CCC(C)(C)OC1 C1(CN(C(c2nc(CC)[nH]n2)C)C)CCCCN1C(c1csc(CC)n1)=O c1(C(N2CCCC2CN(C)C)C(=O)Nc2c(OC)cccc2)nn(C)c(Cl)c1Br C1(NC(C(CC2CCC2)NC(c2c(CC)ncnc2)=O)=O)CCCCC12CC2 C1(C(=O)NC(C)CNC(C2Cc3cscc3C2)=O)CC2(CO1)CC(F)(F)C2 N1(C(C(C#C)(C)C)=O)CC(C(N2CC(CO)C(O)C2)=O)OC(C)C1 C1(C(=O)NC(CNC(c2cccc(C(C)=O)c2)=O)C(C)(C)C)CCCCC1(F)F N1(C(C2(CNC(=O)C(C)COC(C)=O)CC(=C)C2)=O)CCCC12CCOC2 N1(C(CCc2nc(C)sc2)=O)CCC(C)C(CNC(=O)C(F)F)C1 C(c1cccc([N+](=O)[O-])c1)=CC(=O)NCCN(C(C(C(COC)C)C)=O)C n1(CCOCCC)c(N2CCC(CC3CCCCC3)C2)nnc1-c1ccc(C)o1 Cc1[nH]c2ccccc2c1C(N1CCC1CNC(=O)CCc1cn[nH]c1)=O c1(SCc2ccc(C(=O)OCc3nnc(C)o3)o2)ccc(Br)cc1 N1(C(CCNC(=O)OCC)=O)CC2CCN(C(=O)CCC3CC3(F)F)CC2C1 c1(NC(CC2C3CN(C(CNC(N)=O)=O)CC32)=O)ccc2nncn2c1 CC1C(NC(c2ccc(C(N)=O)cc2)=O)CCCN1c1ncc(Cl)c(O)n1 c1(CN2C(CCC(=O)NCCSC)CCC2)n[nH]c2ccc(Cl)cc12 CCCCCCCCCCC(=O)N1CCCC(C)(C)C1CNC(=O)CC(=O)OC N1(C(CC2CCN(C3CCN(C(C(C)=O)=O)CC3)C2)=O)CCc2nnnn2CC1 C1(OC)CN(C(c2ccc(C3CC3CO)cc2)=O)CC1NC(=O)CO.C1CCCC1 Cc1nc(CC(=O)NC2(C)CC(NC(C3CCCN3CC(C)C)=O)C2)cs1 N1(C(c2ccc(OC)c(F)c2)=O)CCCN(C(C2NC(=O)CC2C)=O)CCC1 CCC(CC)CCCC(=O)N1CCCCCC1C(=O)NC(Cc1cnc[nH]1)CO C1(CNC(CSC)=O)CC2CCC1N2C(=O)CN(C1CC1)CC c1(C(N2CCN(C(CC(C=C)C)=O)C(CF)C2)=O)sc2cc(C)cc(C)c2c1Cl C(=O)(C(C)(O)C(F)(F)F)N1CC(CNC(CN(C(C)C)C)=O)OCC1 c1(NC(C2C(CNC(C(COC(C)C)(C)C)=O)OCC2)=O)ccc2occc2c1 N1(C(CSCCN(C)C)=O)CCN(C(=O)C=Cc2cnccn2)C(C(C)(C)C)C1 c1(OCC(=O)NCC2C(NC(C3(C4CCCC4)CC3)=O)C2)ccc(F)cc1 C1(CNC(C(C)(C)CF)=O)CN(C(c2ccc(Br)c(N)c2)=O)CC12CC2 CC1(O)CCCN(C(C23CCN(C(C4(F)CCCCC4)=O)CCC2C3)=O)CC1 C(=O)(CC(F)(F)C(F)(F)F)N1CCC(NC(c2ccc(C)nn2)=O)CC1C CC1CN(C(C2(NC(=O)Cc3ccc(F)cc3)CC(CO)C2)=O)C(C)C1C C1(C(=O)NCC2CCC2CO)CC2CN(C(C34CCCN(CC3)C4)=O)CC2C1 C1(C(=O)NCC2(NC(C(CN(CC)CC)F)=O)CCOC2)CN(S(N)(=O)=O)C1 C1(C(=O)NCC(CC)(CC)CO)CC12CCN(C(C1(Cl)CC1)=O)CC2 N1(C(c2cnccc2-c2cc(C3CC3)cnc2F)=O)CCCC2(CCNC2=O)C1 C1(CC(=O)NC(C(C)NC(C(C)NC(=O)OC)=O)CO)CCN(C(C)=O)CC1 C(=O)(C(C)(C)C1=CCSCC1)N(CC(C)NC(c1cnc(OC)nc1)=O)CC N1(C(C(CC=C)CC=C)=O)CC2(C1)CN(C(C1(C)C=CCC1)=O)CCO2 c1(C(=O)NCCCCNC(C2CC2c2ccco2)=O)cc2cccnc2[nH]1 C1(CCCC)CN(C(=O)C(C)n2ccnc2)CCN1C(=O)CSc1cn[nH]c1 C12(NC(c3occc3C3CC3)=O)CCCC1N(C(=O)CCNSC(F)F)CC2 C1(NC(Cc2c(C)con2)=O)CCSC12CN(C(=O)C(C)CS(C)(=O)=O)C2 Cc1ccc(C(c2nnnn2CC(F)F)NCc2cscc2Cl)c(C)c1 C1(NC(c2c(C)con2)=O)CC(C)N(C(c2cccc(NC(C)(C)C)c2)=O)C1 C1(C(=O)NC(C(=O)NC)CC2CC2)CC(C)CN(C(c2ccc(O)nc2)=O)C1 CC1=C(C(=O)N2CCC(C(=O)NC3CC=CCC3)C23CC3)CCO1 c1(C(=O)NCCC2(NC(=O)C(F)C3CCCC3)CC2)cccc2ccnn12 Cc1cn2cc(C(N3CC4(CCC4NC(c4cnccn4)=O)C3)=O)sc2n1 C1(CCN(C)C(c2ccc(F)s2)=O)CCCCN1C(=O)Cc1cn(C)nn1 Cc1nn(C)c2c(NC3CCC(C)C3)nc(N(C)CC34CCCN3CCC4)nc12 c1(C(=O)NC2CC(CNC(C3CC3(F)Cl)=O)C2)cc2ccccc2nc1O c1(OC)c(C(=O)NC2CC(NC(=O)C(C)n3ccnn3)C2)cc(Cl)cc1Cl N1(C(C(CSC)C)=O)CC(N(C(=O)C2=CCCCO2)C)C(C)(C)C1 N1(C(CNC(C)=O)=O)CCC2CN(C(c3cc(F)c(F)cc3N)=O)CC2CC1 Cc1nc(CN2CCCC2c2ccccc2)sc1-c1nn[nH]n1 Cc1coc(C(C)(C)C)c1C(N1CCCC(CNC(=O)Cc2n[nH]c(=N)s2)C1)=O Cc1cc(C(=O)NCCC2CCN(C(C3CCS(=O)(=O)N3)=O)C2)c(O)nn1 c1(C(CSC)(C)NCCCn2ccnn2)nnnn1CCC1(C)CC1 N1(C(c2ccc(OCC)nn2)=O)CC2COCCC2(NC(=O)C(C)=C2CC2)C1 C(=O)(C(CCSC)NC(N)=O)NCCC1(NC(CCC=CC)=O)CCC1 C(C(C)(O)CC(=O)N1CC(NC(c2cccnc2C)=O)C(n2cccn2)C1)OC Cc1nnc2n1CCC(C(=O)NC(C)CCCNC(=O)CCc1cn[nH]c1)C2 Cc1cc(C(c2nnnn2C2(C)CC2)NCC2(CS(C)(=O)=O)CCC2)cc(C)n1 N1(C(C2(OC)CCC2)=O)CC2CCCC(CNC(=O)C(C)CC3CCC3)C2C1 c1(N2CCC(C)(NC(=O)C=Cc3ccc(Cl)s3)C2)ncnc2ccc(Cl)cc12 c1(CNC(c2nnc(C(C)C)s2)=O)ccc(CNC(C2CC2C2CC2C)=O)cc1 CCC(O)C(C)C(=O)N1CCN(C(=O)CC(C)(C)CC)C(CC(=O)NC)C1 CC1CN2CCN1C(C(N1CC(N(C)C)C(CNC(c3cnc[nH]3)=O)C1)=O)C2 CCCC(CNC(c1csnn1)=O)C(=O)N1CCCN(C2CC2)CC1 C12(NC(C3CN(C)C(=O)C3)=O)CCCC1N(c1ncncc1I)CCC2 C#CCCCCCC(=O)N1CC2CCC1C(NC(c1cn(C)nc1CC)=O)C2 CCCCCCCCC(C)C(=O)N1CC2COCC(C1)C2NC(C1CCC1)=O C1(C(=O)NCC2CCN(C(c3c(C)n(C(C)C)nc3)=O)C2)Cc2ccccc2N1 C1(NC(C)(C)C)CCN(C(=O)C(=O)NC2CCN(C3CCCC3)C2=O)CC1 c1(C(C(=O)NCC(CC=C)NC(c2scnc2Cl)=O)(C)OC)cc(F)cc(F)c1 c1(C(=O)NCC2CN(C(c3c(C)con3)=O)CC2O)cccc2ncsc12 c1(OC)cc(CN2CCN(C(=O)Nc3ccc(Br)cc3)CC2)c(Cl)cn1 Cc1cc(C(=O)N(C(C)CNC(=O)CCCCCF)C)cc(C)c1 c1(C(=O)NCCC(C)NC(c2cnc(C(C)OC)s2)=O)ccc2n[nH]cc2c1Cl C12(NC(CCS(C)(=O)=O)=O)CC(CN=c3cc(C(N)=O)nc[nH]3)(C1)OC21COC1 C(=O)(CC(O)C(C)(C)C)NCCCCCCN(C)C(c1cccc(C(N)=O)n1)=O c1(C(=O)OC2(OC)CC(COC)C2)ccc2ncc(C#N)c-2nc1C(C)C N1(C(c2cnc(CCC)s2)=O)CCC2C(NC(c3c(C)nn(C)c3F)=O)CC12 C1(CC(=O)NCCC2CCCN(C(=O)CC3CSCCS3)C2)COCCOC1 C1(CNC(C2CN(C)C(=O)N2)=O)C2CCC(C2)N1C(c1ccc(C(F)(F)F)s1)=O Cc1cccc(C(=O)NCC2CCC(C)CN2C(=O)CC23COCC(C2)C3)c1O C(=O)(CC(C)(C)N(C)C(C1SCC=C1C)=O)N1CCC(C(=O)NC)C1 N1(C(C(C(CC)CC)C)=O)Cc2ccnn2CC(NC(c2cnsc2C)=O)C1 C1(CNC(c2c(N(C)C)cccn2)=O)CN(C(=O)CCC2OCCO2)CC(C)(C)C1 C=CCC(C(=O)NC1(CC=C)CCN(C(C2CN(C(C)=O)C2)=O)C1)NS(C)(=O)=O C(=O)(C(CCC(C)C)NC(=O)C(F)C(CC)CC)NCCCCCCC=C c1(CC(N2CCC(CCNC(C3(CN(C)C)CC3)=O)C2)=O)ccccc1S(C)=O c1(CC)cc(CNC(c2conc2C(C)NC(=O)CC2CCCN2C)=O)no1 Cc1cc(Cl)cc(C)c1OCC(=O)NC1CC(F)CN(C(c2nn[nH]c2Cl)=O)C1 c1(N2CC(O)(C(C)NC(c3cnc(C)s3)=O)C2)nc2cccc(Br)c2o1 c1(NC(C(C)NC(=O)CC2CCOC2=O)=O)cnccc1C1OCCO1 C#CCCCC(C(=O)NC1COC1)N(C1CCC1)C CS(C)(=O)=Nc1ccc(C(COC(C2CCCOCC2)=O)=O)s1 C1(C(N2CCNC(c3ccccn3)C2)=O)OCCOC1C(F)(F)F c1(NC2CC(CN(C)C)C2)ccc(S(=O)(=O)N2CCC3(C2)CC3(F)F)cc1Cl N1(C(C=CC=CCC)=O)CC(O)(C(C)NC(c2cc(CN(C)C)on2)=O)C1 C(CC1=CCN(C(=O)C(C)O)CC1)NC(c1cc(C)c(C(F)F)cc1)=O Cc1cnc(C(=O)NC2CN(C(=O)Cc3cccc(F)c3)CC2O)cc1Br C(CCCC(c1ccccc1)NC(=O)C(C)OCCN(C)C)OC c1(C(=O)NC2CC3CN(C(c4nnn(CC)c4C)=O)CC32)snc2ccccc12 c1(CC(N2CCC(n3cc(Br)cn3)C2)=O)ncc(C(F)(F)F)s1 c1(NC(C2CN(C(c3cccc(NS(C)(=O)=O)c3)=O)C2)=O)cc(Cl)c(F)cc1Cl C(=O)(C(CC(F)F)N(C)C)N(C)CC1N(C(C2C(C(C)C)CCO2)=O)CCCC1 C1(C(=O)NCC2COCCN2C(c2cc(CCO)on2)=O)CCC=CCCC1 C1(C(=O)NCc2ccc(SC)s2)CCCC(NC(=O)CCN2CCOCC2)C1 c1(CCC(=O)NC(C(C)NC(=O)CS(C)(=O)=O)C)cc2ccccc2o1 C(=O)(C(C(C)CC)N(C(=O)C(CC1CCC1)OC)C)NCC(=O)NCCC CCC(CC(=O)NC(CN(C)C)C(=O)N(C1CC2CCC1O2)C)C(F)F C12(NC(=O)C=CC3CCCCC3)CC3CCC(C1C2)N3C(C1CCO1)=O c1(CNC(C(N2C(=O)CCC2=O)CC)=O)cc2n(n1)CCN(C(=O)CCF)C2 C1(C(=O)NC23CC(NC(C(C=C)CC)=O)(C2)C3)Cc2nnc(C)n2C1 c1(C(=O)NCC2CC3(CN(C(c4[nH]c(=N)sc4)=O)C3)C2)cnc2c(c1)CCCO2 C1(CCOC)(NC(=O)Cc2nc[nH]n2)CCN(C(=O)C(C(C)C)n2cncn2)C1 C(N=C(NCC(C)(C)C)N1CCC(OC(F)F)C1)c1c(OC)cc(C#N)cc1 C#CCC(C)(C(=O)NC1(C)CCC(C)C1)NC(C1CC(C)(O)C1)=O c1(C(N2CC(NC(c3c(CC)n(C)nc3)=O)C(OC)C2)=O)nc(C)c(C)[nH]c1=O C(=O)(C(CCC(N)=O)N(C)C)NCCCCN(C(C(Cn1ccc(C)n1)C)=O)C CCCC(O)(CCC)CC(=O)NC(C)C(C)NC(c1cccc(O)c1Cl)=O Cc1cn2cc(CC(N3CC(CNC(=O)C=Cc4cnc[nH]4)CC3C)=O)nc2s1 c12cccc(c1)NC(=O)CC2.C1(CCC#C)CCCN1C(C)=O N1(C(C=C(C)C2CC2)=O)CCC2CCN(C(=O)CSCc3ccccc3Cl)CC12 C1(C(N(C2CCN(C(c3cnc(O)o3)=O)C2)CC)=O)CCCCC1(C)C c1(CC)ccc(C(=O)NC(CN(C)C)C(=O)N2CCC(n3ccnn3)C2)o1 Cc1cc(NC(CNC(c2cnoc2-c2ccco2)=O)C(C)(C)C)ncn1 O=C(CCCCCBr)NC1CCCN(C(=O)CCc2cccc(OC(F)F)c2)CC1 c1(C(C)(C)C)nccc(=NC(=O)C2CCC(CC(=O)Nc3n[nH]cc3I)CC2)[nH]1 c1(OC2(C(N(C3CCN(C(C(CC)OC)=O)C3)CC)=O)CC2)cccc(C)c1C C#CCC(C(=O)OC)NC(=O)CN(C(=O)Cc1cncc(C)c1)C(C)C C1(N(c2cccc(CO)c2)C(=O)NCC(=O)OC)CCNCCC1C c1(C(=O)NC23CCN(C(C=COCC)=O)CC2C3)cnc2onc(C3CC3)c2c1 N1(C(c2n(CC)ccn2)=O)CC(NC(C2CN(CC3CCCCC3)C2)=O)C2CC12 c1(OCC(=O)N(CC(C)(C)NC(C2CCC2)=O)C)cc(Br)ccc1F C1(F)(N(CC(C)(C)C)C)CCC(=O)NC1=O C1(CNC(CC(CNC(CCOCCOCC)=O)OC)=O)CCC=CCCC1 CC(O)CCCC(=O)NC(CNC(=O)C(C)(C)Cc1ccccc1)C(C)C C(=O)(C1=C(C)N2CCN=C2S1)NCC(CC)(CC)CC c1(CNC(c2n(CC)nnn2)c2ccsc2Br)cccc(CC(=O)OC)c1 C=CCC(CC(C)C)C(=O)NCCOC1CN(C(=O)CCC(C)CN(C)C)C1 CC(C)CCC(=O)C(=O)N1CCN(C(=O)Cc2ccc(C(F)F)cc2)CC1C N1(C(C(C)(C)SC)=O)CC2CC(C(=O)N(C)CCc3cccs3)C(C2)C1 c1(CN2CCC(N(C)C(C3(c4ccsc4)CC3)=O)C2)cnn(-c2ccccc2)c1N C1(C(C(=O)C=CC2CCN(C(=O)CN3CC4CC4C3)CC2)=O)CC2(C1)CC(CO)C2 C1(N(C(CC=CC)=O)C)CN(C(C2CC2F)=O)CC1(C)C n1(CC)cc(CC(=O)NCCC2CCCN2C(c2cn(C(C)C)cn2)=O)cn1 C1(COC)CN(C(=O)COCCF)CCN1C(c1cn(C(C)C)cc1C)=O c1(CN2CCCC(C(N3CC(C)C(=O)CC3)=O)CC2)cc(F)c(Cl)c(Cl)c1 C(=O)(CCCCC#N)NCC(C)NC(=O)C=CC(c1cnn(C)c1)=O c1(CC(C(=O)NCCC2C(C)CN(C(c3ccco3)=O)C2)O)c(F)cccc1Cl N1(C(C2(C(C)(C)OC)CC2)=O)CCC(C(C)(C)NC(=O)CCCSC)C1 C(C(CO)(CO)NC(C1CCC1c1nc(S)n[nH]1)=O)N(C)C(C1CCCC1O)=O CC1(C)CCN(CCNC(=O)C(c2cccnc2)NC(=O)C(F)=CC2CC2)C1 c1(C(N2C(CNC(C3CC4CCC3C4)=O)CCC2)=O)cc2n(n1)CCO2 CCC(C)(O)C(=O)N1CCC(C2CCCN2C(=O)C(CCCS(N)(=O)=O)NC)C1 C1(C(=O)NCCC(C)(C)NC(C(C)=C(C)C)=O)Cc2n[nH]cc2C(=O)N1 CC(O)CC(C)(C)CNC(=O)C=CC(C)NC(=O)Cc1ccc(O)cn1 N1(C(CC(C(C)C)c2ccccc2)=O)CC2CCN(C(=O)C(C)(C)C#N)CC2C1 C1(C(=O)NC(CNC(c2cnc(CC)[nH]2)=O)(C)C)CCC(=O)N(CC)C1 C1(N(CCOC)C)CCCCC1CNC(C1C=CCN1C(=O)OC(C)(C)C)=O CC1CCCCC1(CNC(C1CCCN1C=O)=O)NC(=O)CC(C)n1ccnc1 Cc1cn2cc(CC(=O)NC3(CNC(C4(C)CCOC4C)=O)CCCC3)nc2s1 CCCC(C)(O)C(=O)NC1CC(C)CN(C(C2(CO)CC2)=O)C1 N1(C(CN(C(=O)OC)C)=O)CCCC2(CCCCC2NC(c2cc(C)cs2)=O)C1 C(=O)(CCC(=O)c1cc(C)sc1C)NC(CC=C)CNC(=O)C(C)(C)OC(C)C C1(NC(CC(=C=C)C)=O)CN(C(=O)C(C)OCC(C)C)CC12CCOCC2 C=CC1COCCN1C(=O)CC(C)NC(c1oc(C)nc1C)=O C1(C(=O)NCC2(F)CCN(C(=O)Cc3ccsn3)CC2)CC2C=CCC(C1)C2 c1(C(N2CCC(NC(C(N)=O)=O)C(CO)CC2)=O)ccc2c(c1)CCCS2(=O)=O CN1CCC(=CC(=O)NCC(F)CNC(=O)Cc2cnc(C(C)(C)C)[nH]2)CC1 c1(C(N2CC(NC(=O)NC)C2)=O)coc(CNC(=O)CC2CCOC2C)n1 N1(S(CC)(=O)=O)CCc2ccc(CNC(c3cccc(N(C)C)n3)=O)cc2C1 c1(C(=O)NCC2CCCN(C(C=CC)=O)C2)cccc2c1CCCC2=O N1(C(c2c(C(C)C)con2)=O)CCC2(CO)CN(C(c3cnc(S)[nH]3)=O)CC2C1 N1(C(C2CC(C)(C(=O)OC)C2)=O)CCCC(O)(CNC(c2ccccn2)=O)C1 N1(C(c2c(C)csn2)=O)CC(CC(=O)NCc2cnc(O)c(F)c2)CC1(C)C C12(CNC(COCC(C)C)=O)CCCC1N(C(c1ccc(C#N)cn1)=O)CCC2 N1(C(c2c(C)scn2)C(=O)NCCC2CC2)CCC2(CC1)COCC(=O)N2 Cc1ccc(O)c(C(=O)NCC2(NC(C3CN(C(C)C)C3)=O)CCOC2)n1 c1(NCCC2C(C)CCCN2C(=O)C2=CCCCO2)ncnc2cccnc12 C1(=CCNC(C2C(C)CCO2)=O)CCN(C(=O)C(F)(F)CO)CC1 N1(CC(=O)NC2CCCCC2)CCN(Cc2ccncc2Cl)c2c(F)cccc21 C1(C(=O)NCCCc2n(C)ncc2)CC1C1CN(C(=O)CN2CC=CC2)C1 C12(NC(c3ccc(CC)[nH]3)=O)CCCC1N(C(c1snc(Cl)c1Cl)=O)CCC2 C1(C(=O)NC2CCC(NC(C3(CO)CCCCC3)=O)C2)CC12CCSCC2 C(=O)(C1=CNC2=NCCCN12)N1C(CCNC(C2CC(OC)C2)=O)CSCC1 C(=O)(C(O)CC(F)(F)F)N1CCC(OCCNC(C2(N(C)C)CCC2)=O)C1 C1(CNC(=O)CCc2cscn2)CCN(C(=O)CCC2CC2(F)F)C12CC2 C1(CNC(=O)CCOc2cccc(Cl)c2)CN(C(=O)CC=C(Cl)Cl)CCCO1 C=C(C)C(C)(O)C(=O)NC(C)CN(C)C(c1cc2sccc2s1)=O Cc1nc2ccnn2c(C)c1C(=O)NCC(C1CC1)N(C(=O)CC1CCC1)C c1(-n2ncc(NC(=O)NCCn3c(C)cc(C(F)(F)F)n3)c2)ncc(Cl)cc1Cl CN1N=C(CC(=O)NCc2cccc(CNc3ccnc4ncnn34)c2)CC1=O N1(C(COC(CC)C)=O)CCC(CCNC(c2cnn(C)c2COC)=O)CC1 c1(OC)ccc(Cl)cc1CC(=O)NCC(O)CNC(=O)CC1COCCOC1 C1(C(=O)NCCSC(C)C)CCC(CNC(=O)CSC(F)(F)F)C1 C(=O)(C1=C2CCN=C2NC=C1)N1CCN(C(Cc2cc(C)nn2C)=O)CC1C N1(C(c2cccc(C)n2)=O)CCN(C(c2ccn(CCF)n2)=O)CC1CO N1(C(C(COC)(F)F)=O)Cc2ccccc2C(NC(=O)CN(C)C)C1 C(=O)(C(F)CC(CC)CC)NC(CNC(CC(CC=C)(C)C)=O)(CC)CC Cc1nc(CO)sc1C(=O)N(CCCNC(=O)C=Cc1cccnc1)C(C)C C(c1cc(C)no1)=CC(=O)NC1CC(CNC(c2c(CCC)nco2)=O)C1 C=CC1(C(=O)NCC2=NOC(C)C2)CCN(C(C2CC23CCCC3)=O)C1 C1(C(=O)Nc2c(C(=O)OC)cc[nH]2)CCC(C)N(C(C2CC2C(F)F)=O)C1 C1(C(=O)NC2(CC)CN(C(=O)CC(C)OC)C2)CC12CCCC2 c1(CC)nn(C)c(C(c2nnnn2C(C)C(=O)OC)Nc2ncoc2C)c1Cl c1(C(N2CCC(N(C(c3cn(C)c(=O)cn3)=O)CC)C2)=O)ncc([N+](=O)[O-])n1C N1(Cc2c(C)nc[nH]2)CCCN(C(c2ccc(Br)c(C#N)c2)=O)C(C)C1 c1(NC(c2cn(CC)nc2)C)cc(=NC2CCN(CCOC)C2)[nH]c(COC)n1 c1cnc2c(=NCCc3ccoc3)[nH]c(N3CC4COCC(C4)C3)nc2c1 S(=O)(=O)(c1c[nH]c(=NCCCS(=O)(=O)CC)cc1C)NCC(CC)N1CCCC1 N1(C(C2C(C)(CC)C2)=O)CC2(CCC(NC(c3nc(C)c(C)[nH]3)=O)CC2)C1 C(C)(CCC(=O)N1CCN(C2CN(C(=O)CCCOC)C2)CC1)OCC.C(C)COC C(=O)(C(C)(C)O)N1C(C(=O)NCCNC(COC)=O)CC1 c1(C(=O)NCCNC(C(C)(C)c2ccsc2)=O)cc(S(N)(=O)=O)c[nH]1.C12CN(C1)C2 N1(C(c2ncccc2F)C(=O)NCCCSC)CCC2(CCCC2)C1 c1(C(=O)NCC(CC=C)NC(=O)C(O)C(F)(F)F)ccc2c[nH]nc2n1 C(=O)(CS(=O)(=O)CC)NC(C(=O)NCC(CCCC)O)Cn1cccn1 N1(C(C(C(C)O)C)=O)CCCC(C)(C)C1CNC(C1CC=CCO1)=O C1(CC(=O)NCC(CC)N(C(=O)CCC=CC(C)C)C)C=CCCC1 c1(C(=O)NC2CN(C(c3nc(C)[nH]n3)=O)CC2C)cccc2c1C(=O)NC2=O c1(CN2CCC(CC(=O)NC(c3nn[nH]n3)CC)C2)cccc2c1ccn2C N1(CCN(C(=O)Cc2cnn(C)c2C(F)(F)F)C)CCN(C(C2(F)CC2)=O)CC1 c1(NC)ccc(C(=O)NCC2CC(F)CN2C(=O)CCCc2nc(C)no2)cc1 N1(C(COCCC#C)=O)CCCC(C(=O)NC(COC(C)=O)CO)C1 CC1(C)CCC(C(=O)NCC2(F)CCCC2)CN1C(=O)Cn1nccn1 c1(C(=O)NC(C(C)NC(Cc2cc(C)on2)=O)C)cccc2ncnn12 CC1CN(C(=O)C(O)CC2CCCC2)CCC1NC(=O)CCNC1CC1 c1(CC)ncccc1C(=O)NCCC1(NC(=O)CSC)CC1 Cc1ccc(C)c(C(=O)NC2CC(c3n[nH]c(=N)o3)C2)c1O C1(C(=O)NCC(COC)(F)F)(CF)CCN(C(c2ccccc2C2CC2)=O)C1 C(CC(C)C(=O)NCC(C)(C(C)C)NC(c1cc(C)c(C)s1)=O)=CC N1(C(C2(OC)CCOCC2)=O)CCCC(CO)(NC(C2CCC(=O)NC2)=O)C1 C(=O)(C1=CC2C=CC(C1)C2)NC1C(CNC(c2c(Cl)ccc(OC)n2)=O)CC1 c1(CCCC)nc(C(=O)N(C)CCN(C)C(C2CCC(C)C2)=O)cs1 Cn1c(C(=O)NCCN(C(c2cn(C3CCOC3)cn2)=O)C2CC2)cnc1O CN1CC2CN(C(=O)C(=O)NC3CCCCC3C(F)(F)F)CC2(C)C1 C(C(C(=O)N1CCC(O)(C(F)F)C1)C(C)(C)C)NC(Cn1nnc(C)n1)=O Cc1cc(C(=O)NC(C)CCCNC(=O)Cc2cnccc2Cl)n(C2CC2)n1 C1(NC(C2(C=C)CCC2)=O)CC2CC1N(C(=O)C(C)Oc1cccc(C)c1C)C2 C1(C(=O)NCCNC(C)=O)CC(C)N(C(c2nnn(C)c2C)=O)C1 c1(C(N2CCC3(CN(C(C(C=C)O)=O)C3)C2)=O)c(C)nn2cccnc12 CCC(CNC(c1ccccc1C(F)F)c1nnnn1C1(C)CC1)CCCO C12(NC(c3ccc(F)cn3)=O)CCC(NC(C3CN4CCC3C4)=O)(CC1)C2 c1(C(N2CCCC(C)(OC)CC2)=O)ccc2c(c1)CCC2(F)F c1(OC)cccc(C(N2CC3C(C2)C3(F)F)C(=O)NCC2CC2)c1C c1(CC)ccc(C(=O)NC23COC(CNC(C4CCOCC4)=O)(C2)C3)cc1Cl C1(C(=O)NC(c2ccco2)COC)CCC(NCc2cc(C)n(C)n2)CC1 C(CN=c1cc(C)nc(NC2CCC(c3cccc(C)n3)C2)[nH]1)OCC.C12CC1C2 n1(CCC(=O)NCCC(C)NC(C(COC)CC(C)C)=O)cc([N+](=O)[O-])nc1C C1(C(N2C(C)CCC2(C)C)=O)CCN(C(=O)CC2CCC2)C(C)(C)C1 C1(OC)CN(C(=O)C(C(C)C)NS(C)(=O)=O)CC1CNC(=O)CC1CC(F)C1 C12(NC(c3c(CC)ccc(C)c3)=O)CCCC1CN(C(=O)C=CSC)C2 C1(CN(CC(c2cc(F)ccc2F)=O)CC)CC2(CO1)CC(F)(F)C2 N1(C(c2ccc(C)s2)=O)CC2CC(C1)C(CO)C2NC(C1CC(NC2CC2)C1)=O C1(CC(N2C(CN(C(C3(C)CC(=C)C3)=O)C)CCC2)=O)CCS(=O)(=O)C1 c1(OC)cccc(-c2nc(CC3CCSC3)n(C(C3CCC3)C)n2)n1 N1(C2CCN(C(C3CC34CCC4)=O)C2)CCN(CCC(N2CCCCC2)=O)CC1 c1(OC)nc(C)ncc1C(=O)NC1CCCCN(C(c2cnc(C)[nH]2)=O)C1 CCCCC(CCCC)C(=O)NCCCCCCN(C)C(C1C2CC3C(C2)C13)=O CCS(=O)CC(=O)N1CCCCC1CNC(=O)Cc1coc(C)n1 C=CCCCCCCC(=O)N1CC(OC)C(NC(C2(O)CCCC(C)(C)C2)=O)C1 C(=O)(C(C)(C)C1=CCN(C(c2cccnn2)=O)C1)NC(CC(C)(C)C)CO C(CN=C(NCCNC1CCC1)NCC(C)NS(C)(=O)=O)c1ccc(OC)cc1 C1(NC(c2c(NC(C)=O)cccn2)=O)CN(C(c2n[nH]c(C)c2O)=O)CCC1C C=CC(C)(O)CC(=O)N1CCC(NC(=O)C(C)NC(=O)NC(C)C)CC1 Cn1ncc2cc(C(=O)NCC3CC(NC(C4(C)COC4)=O)C3)sc12 C1(C(=O)NC(C=C)C)CC2(CC(NC(c3ccc(Br)c(OC(C)C)c3)=O)C2)C1 CC(C)(Cc1ccccc1)C(=O)NCC1C2CN(C(C3(Br)CC3)=O)CC12 C(CCNC(=O)CCSCC(C)C)(C(C)C)NC(c1nc(C(C)OC)sc1)=O c1(C(=O)NC2CCCC(CNC(C(C)SCC)=O)C2)ccc(C)nc1O c1(-c2cc(C)c(F)cc2)ccc2sc(C(=O)Nc3c(C#N)cnn3C)cc2c1 c1(C(N2CCCC(NC(C(C)(C)c3cccnc3)=O)C2)=O)cc(Cl)c(F)cc1N N1(C(CC(COC)COC)=O)C(C)CC2CN(C(c3cc(N)cc(F)c3)=O)CC12 C(=O)(CC1=NN(C)C(=O)C1)NC(C1CCCN(C(=O)C=CC2CCOCC2)C1)C C1(CNC(c2cnc3n2CCC3)=O)CN(C(=O)C(F)CC2CCC2)C2(CCC2)C1 CCC(CC)(CCNC(=O)C(C)Cn1ccnc1)NC(=O)C(C)CF c1(OC(CC)C)cc(CN2CCC(C)(C(=O)NC3CC(F)(F)C3)C2)cc(Cl)c1 Cc1ccoc1C(=O)NC(CC1CC1)C(=O)NCC(O)Cn1cccn1 C1(=O)C(C)(C)C(=O)NCC(CC=C)N1.c1(C(=O)OC(C)(C)C)ncsc1C CC1CN(C(=O)C(C)(C)F)CC(C)CN1C(C1CCCN(C)C1)=O C(=O)(C1CCCc2nncn21)NC(C1(O)CN(C(c2ccc(C#C)cc2)=O)C1)C C1(C(N(CC(=O)Nc2ccc(O)cc2F)CC#C)=O)Cc2ccccc2C1 c1(C(=O)NCCCC(C)NC(c2c(NCC)scn2)=O)c(Cl)c([N+](=O)[O-])nn1C N1(CCc2c(OC)cccc2OC)C(=O)NC2(CCc3ccccc3C2)C1=O C1(CCCNC(C(CN(C)C)O)=O)CN(C(=O)CC2(C)CC2)CCO1 C(C)(C(C(=O)NCc1ccnc(O)c1)NC(C1COCCC1C)=O)OC N1(C(C#CCNC(C(C(=O)OC)(C)C)=O)=O)CC2COCC(C2)C1 Cc1cn2cc(C(=O)NC3CN(C(=O)CCC4CCC(C)O4)C3)cc(C)c2n1 c1(C(=O)NCC(CNC(C2(COC)CCC2)=O)OC)cccn(CC2CC2)c1=O CC(C(=O)N(CC(C)(C)NC(c1cnc(C2CC2)nc1O)=O)C)C(F)(F)C(F)F CN(C)NC(=O)CCC(=O)N1CC(CNC(C2(O)CC2)=O)N2CCC1C2 c1(C(N2CC(CCCCNC(C3N(CC)CCC3)=O)C2)=O)cc(C#N)n(C)n1 CC1(NC2OCCC2C(=O)NS(C)(=O)=O)CCN(C(=O)CN2CCOCC2)C1 c1(OC)cc(C(=O)NCC2CCCC2NC(=O)CC(O)CC2CC2)ncn1 C(=O)(C(=O)N=c1nc2n([nH]1)CCCC2)Nc1c(C(=O)OCC)c(Cl)ccc1 Cc1cccc2cc(C(=O)NCC(CO)NC(c3cc(C#N)ccc3Cl)=O)nn12 CC(F)(F)C(F)C(=O)NC1CCCC1CC(=O)NCCCN=[N+]=[N-] c1(C(N2CC3C(NC(c4cc(F)n[nH]4)=O)C(C3)C2)=O)ccc2cnccc2c1 c1(CN2C(CC)CN(C(c3ccon3)=O)CC2)ccc(C#N)cc1S(C)(=O)=O C1(N(C(=O)C=CC2CCOCC2)C)CN(C(=O)C(F)OC(F)(F)F)CC12CC2 Cc1ccc(CCC(=O)NC2CC(NC(=O)C(Cl)=CCl)C2)c(Br)c1 c1(NC(C2N(C(CC(C(C)C)O)=O)CCCC2)C)cccc(F)c1C#N c1(NCCC(=O)NCCC2CN(C(C(C)(C3(C)CC3)OC)=O)C2)ccccc1C C1(C(=O)NCC(CC=C)NC(c2cnnn2C)=O)CCN(S(N)(=O)=O)CC1 C(=O)(C#CC(C)(C)C)NCC1CCC(C(N(C)Cc2ccc(O)cc2)=O)O1 c1(CCC(=O)NCC2(NC(c3ccc(C)cn3)=O)CC2)ccc(F)cc1Cl C=CCCN=C1NCCC(C(C)(C)C)C(CCCCC)CC(CO)CN1 C(N=c1[nH]c(Cl)ncc1CC)C1N(C(c2n(C=C)ncc2)=O)CCCC1C c1(CC)ccc(C(N2CC(NC(c3ccc(C#N)[nH]3)=O)CCC2C)=O)c(C)n1 C(=O)(C(=O)N=S(C)(C)=O)NC1C(NC(C2(C)CN(C)C(=O)C2)=O)CC1 N1(C(C2CN(C(=O)C3CC3)CC2C2CC2)=O)CCc2c(O)noc2C1 N1(C(Cc2ccc(C)nc2)=O)CCCC2(NC(=O)C(F)C3CCC3)CC2C1 c1(CC(=O)NC2C(C(N(CCCO)CC)=O)CCC2)cccnc1O C1(C2CCCN(C(=O)C(C)(C)n3ccnn3)C2)(NC(C2CC(C)C2)=O)CC1 N1(C(CCCOCCOC)=O)CC2CC2(CNC(=O)CC2CCCO2)C1 CC(C)(CC1CC1)C(=O)N1CCCC1C(N1CC(O)(C(N)=O)C1)=O N1(C(c2cnn(CCF)c2)=O)CCCC2(C1)CN(C(c1ccco1)=O)CCO2 N#CCCCC(=O)NCCOC1CCN(C(C2(n3cc(Br)cn3)CC2)=O)C1 c1(CC(=O)NCCCCC(C)NC(C2(C)CC2)=O)cc(Br)ccc1F N1(C(C=CCCC)=O)CCC(NC(=O)CC2CCOC2(C)C)C12CC2 c1(CC(=O)NCC2C(NC(CC=C(C)C)=O)CCC2)cnc2ncccn12 C(C(C)C)(C(O)C(=O)N1CC(CCNC(C2CC23CCC3)=O)C(C)C1)OC C(N=c1[nH]c(C)cc(=NCC(C)(C)SCCO)[nH]1)c1ccn(CCC)n1 N1(C(CC2(CC)CCC2)=O)CCC(N(C(c2ccccn2)=O)CC)CC1 c1(CNC(C=C(C)C(C)C)=O)ccc(C(=O)N(C)C(C2CCCO2)C)cc1 C1(CNC(C2C(NC(C(C(C)C)OC)=O)C2(C)C)=O)CCCN(C)C1=O N1(C(C)C)CCCC(NC(=O)CCNC(=O)Cc2cc[nH]c2)C1 C1(NC(c2n(CCCOC)nnn2)c2ncc(C)s2)CCCC=C1Br N1(C(CCCN(C(C)C)C)=O)CCC2(CC2C(N2CCC3C(C(N)=O)C3C2)=O)C1 N1(C(C2CCSC2)=O)CC=C(CNC(C23CC4CC2C3C4)=O)CC1 c1(CN2CC3(CCN(C(C(C)(C)O)=O)C3)C2)cc(C(=O)O)cc([N+](=O)[O-])c1 CC(C)(C)C(CC(=O)NC1CN(C(=O)CCF)CC1(C)C)C(F)F C#CCC(C)(C(=O)NCCCOC1CC1)NC(=O)C1=CCCC1 C1(NC(C2C(C(C)C)C2)=O)CC2CCC(C1)N2C(=O)Cc1cnns1 N1(C(c2c(CC)ncs2)=O)Cc2occ(C(=O)NC3CCC(F)(F)C3)c2C1 N1(C(c2n(C(C)C)ccn2)=O)CCN(C(c2cccc(O)n2)=O)C(CF)C1 c1(-c2cn(CC3N(C(C(C=C)(C)C)=O)CCCC3)nn2)cc(OC)c(OC)cc1F c1(C(=O)NC2CC(OCCN(C)C)C2)ncsc1S(N)(=O)=O.c12cn(nn1)C2 c1(OC(F)F)cccc(CNc2csc(C3CCCO3)n2)c1Br C#CC1(C(=O)NCC(c2ccnn2C)O)CCN(C(c2cnco2)=O)C1 C1(C)(C(=O)OC)CCC1(C)C(=O)NCC(C)(C)CN(C(=O)C(F)C1CC1)C C(C(C)(C)CC(F)F)NC(C(C)N(C(c1cc([N+](=O)[O-])n[nH]1)=O)C1CC1)=O N1(C(CN(C(COC)=O)C)=O)CCCC(Cn2cc(COCCO)nn2)C1 Cc1nncc(CNC(C2(NC(=O)C(C)OCC(C)C)CC2(C)C)=O)c1C c1(C(=O)NCC2CCN(C(=O)C=Cc3ncco3)C2)cc2c(s1)CCOC2 c1(C(N(CCNC(CSCC#C)=O)C(C)C)=O)oc2ccccc2c1Cl c1(C(N2CCC(F)(CNC(C(C)SC)=O)CC2)=O)cc(=O)n2nccc2[nH]1 c1(NC(C(N2CC(C(=O)OC)C(C(F)(F)F)C2)=O)=O)c(Br)nc2n1CCOC2 c1(CNC(CNC(CNC(CC2CCC(C)C2)=O)=O)=O)cc(F)cc(F)c1 C1(CNC(C2CSCN2C(C2(CCF)CC(O)C2)=O)=O)CC2CCC1O2 N1(C(c2nccc(OC)c2)=O)CCCC(O)(CNC(C2CC(C(C)C)=NO2)=O)C1 Cc1ccncc1CC(=O)NCCC1(NC(C2CCCO2)=O)CC1 c1(CC(=O)NCC2C(NC(CCNC(=O)C=CCl)=O)C2)ncc(F)cc1F C1(CNC(CCCCNC(C)=O)=O)COC(C)(C)CN1C(=O)C(C)c1ccsc1 N1(C(CCCc2c(C)ccs2)=O)CC2(CCC2NC(=O)C(C)OCCN(C)C)C1 CCCC(C(=O)NCC(CO)NC(c1nn(CC)cc1Cl)=O)C(C)C c1(CC2CCN(C(C3(CCO)CCCCC3)=O)CC2)ccc(F)c(F)c1 c1(C(=O)NC(C)CNC(C2(Cl)CC23CCC3)=O)ccc(P(C)(C)=O)cc1 N1(C(Cc2c(C)nsc2)=O)CCCC(C)(NC(C2CC=CCO2)=O)C1 C(=O)(C(CO)NC(N)=O)N(C1CCN(C(c2csc(-c3ccoc3)n2)=O)C1)CC C1(NC(c2cnc(C)nc2C)=O)CN(C(=O)C(C)CC2CC2)CC1S(C)(=O)=O c1(CNC(C2CCCN2C(=O)CNCc2ncsc2Br)=O)ccc(Cl)nn1 c1(C(=O)NCC2CC(NC(C3(C)CCNC3=O)=O)C2)cccc2cc(O)ccc12 C1(C(=O)NC2CC(NC(c3cc(F)cs3)=O)C2)CCc2ccnn2C1 C(CCCCC(=O)N(CC(C)(C)CNC(c1ccccc1N(C)C)=O)C)SC C1(NC(c2ncn(CC)c2)=O)CC(O)CN(C(c2cc(C3CCC3)[nH]n2)=O)C1 C1(C(=O)N(CC)CC)(NC(COC(CC)CC)=O)CC(F)C1 C(=O)(C1=CCCCO1)N1CC(OCCNC(CC2C(C)=NOC2=O)=O)C1 C1(C(=O)NC2C(OC)CN(C(=O)CC3(C)CC3)C2)(OC)CCCCCC1 c1(N2CC(CC)OCC2)ccc(S(=O)(=O)NC(c2cnc(Cl)s2)C)cc1Cl c1(CC)c(C(=O)NC2(C)CCN(C(=O)CC(O)C3CCCC3)CC2)cccc1C Cc1ccc(C(=O)N(C)CCNC(=O)CN(S(C)(=O)=O)C)c2ccccc12 C1(CCc2scc(C(=O)NOCC3CC3)n2)CCCCC1NC(=O)C=CBr c1(OC)cccc(C(C)CC(=O)N2CC(NC(=O)C(C)C)C2)c1 n1(CC)nc(C(=O)NCCN(C(=O)C(c2cccc(O)c2)(C)C)C2CC2)cc1C C1(C(=O)NCC2CCCN(C(C(C)(C)OC)=O)CC2)Cc2ccccc2N1C C1(c2nc(-c3c(C(=O)OC)n(Cc4ccccc4)nn3)on2)CC2CC(O)C2C1 CC1CCN(C(c2ncc(Cl)s2)=O)C1CNC(C1CC(O)C1)=O C1CCCCCC1.C(CCCCCN)N(C(C)=O)C(c1c(Cl)noc1C)=O CC(C)C(CCNC(=O)C(=O)NC1CC1)NC(=O)C(C)(Cl)Cl c1(C(=O)NC2(C)CC(NC(=O)C=C3CCSCC3)C2)cnc2sccn2c1=O c1(CC(C)C)ccc(C#N)c(N2CC3CC2(NC(=O)C(C)CC(N)=O)C3)n1 C1(C(=O)NCCC(C)NC(=O)CCCc2n[nH]c(=N)s2)CCC(=C2CCC2)CC1 c1(C(N2C(C(=O)NC(CC(C)(C)C)CO)CC3(CC3)C2)=O)cc2ccccn2c1 CC(C(=O)NCCCN(C)C(C1CCSC1)=O)N(C)C(=O)OC(C)(C)C C1(OC)CN(c2nnc(NC(=O)OC(C)(C)C)s2)C(C)(CNC(=O)CCOC)C1 C(N=c1[nH]c(N2CCC(c3cc(O)n[nH]3)C2)nc2c1COCC2)c1nc(C)sn1 c1(CC)cc(Br)ccc1C(=O)Nc1cccnc1C(N1CCC(F)(C(=O)OC)C1)=O CC(C)C(C)(O)C(=O)NCC(C)(C)OCCNC(c1ccc(SCCO)cc1)=O c1(C(N2CC(CNC(C3(CCCC)CCC3)=O)(OC)C2)=O)c(C)cc(C)nc1O CC(C)CC(C)CC(=O)NCc1ncc(C(N2CC3OCC(CO)C3C2)=O)cn1 Cc1c(CC(=O)NC2CN(C(c3cnc(C#N)s3)=O)C2)c(O)nc2[nH]nc(O)c12 c1(COC)ccc(C(=O)NCC(O)CCNC(=O)C(N2CCOC2=O)C)o1 O=C1CCN(C(=O)Cc2cscn2)C2CCN(C(c3ccc(Cl)o3)=O)CC2N1 c1(C(=O)NCCNC(c2cccc(C)c2F)=O)c(C2CC2)nc2sccn12 C(CC(=O)N1CC(NC(C2(C)CCCC2(F)F)=O)C1)(C1=CCCC1)OCC CC1=C(C(=O)NCC(N2CCN(C(=O)C3=CCCC3)CC2)=O)CCO1 N1(C(c2ccc(Br)cn2)C(=O)NCc2ccc(F)cc2)CC2CCCC12 C1(CC(=O)NC(C(=O)NCCC=C=C)CC2CCCC2)CCCC12CC2 Cc1ccc(CC(N2CCOCC(CNC(c3cnccc3C)=O)C2)=O)cc1C C1(CCC)CN(C(C2CCN(C(c3cn(CC)cn3)=O)CC2)=O)CCO1 C1(N(C)CCO)CCN(C(=O)C(CN2CCCC2)c2ccccc2)CC1 C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CCC2CN(C(CCCCCOC)=O)CC21 N1(C(C(C)(C)F)=O)CCC2(CC1)CC(NC(=O)CCN1CCCC1=O)C2 CN1CCN(C(c2cc[n+]([O-])cc2)=O)CC1CNC(c1nccnc1CO)=O Cc1c(C(N2CCC(C)(N3CCOCC3)C2)C(=O)N(CC)CC2CC2)cccc1Br c1(C(=O)NC2(C)CN(C(C(C)CC3CCCO3)=O)C2)cc2ccsc2c(O)n1 c1(NC(=O)Nc2cccc(CC)c2)cc(F)ccc1Oc1cncc(CO)c1 C1(N(C(CC2C(CC)C2)=O)C)CN(C(=O)CCC2CCC(=O)N2)CCC1C N1(C(c2scc(C(N)=O)c2)=O)CCC(NC(c2ccsn2)=O)C1c1ccccc1 N1(C(c2c(OC)c[nH]n2)=O)CC(NC(=O)CC2(O)CCCC2)CC12CCCCC2 Cc1ccc(OCCC(=O)NC2(CNC(c3cnc(C)cn3)=O)CCOC2)cc1 C1(NC(C2C(C(=O)OCC)C2)=O)CC(C)CN(C(c2cc(OC)n(C)n2)=O)C1 C1(C(=O)NCC=CCC(=O)N(c2c(C)cccc2)C)C2CCC(C2)C1C C(=O)(C(C(=O)NCCN(C(c1ccc(C)nn1)=O)Cc1ccccc1)OC)OC C1(C(=O)NCC2CCCC(NC(=O)CCCCN3CCCC3)C2)CC2C(C1)C2(F)F c1(C(N(C2CN(C(=O)CSCc3ccc(F)cc3)C2)C)=O)cn(C)c(=O)nc1O Cc1cccc(C(=O)NCC2CC(O)CN2C(c2ccc(Br)c(O)n2)=O)c1C C1(c2cn(CCC(=O)NC)nn2)N(C(=O)CC2CC(=O)NC2=O)CC12CCC2 C(C(C)C(=O)NCCC12CC(CO1)C2)NC(C(C)N(C(C)=O)C)=O c1(C(=O)NCCCCCNC(C2C(SC)CCC2)=O)cc(C)nn1C(C)(C)C c1(OC)cc(Cl)c(Cl)cc1C(N1CC(NC(=O)C(O)Cn2cncn2)C(O)C1)=O Cc1nc(NC(c2cc(C3CCC3)on2)=O)cc(O)n1.c12cccc(c1)NC2C C(=O)(CN1C(=O)Cc2ccccc21)NC(CN(C(c1cnccc1Cl)=O)CC)C CC(C)(C)C(=O)C(=O)N1CC2(CC2)CC1CNC(C1CC(CC(F)F)C1)=O c1(C(N2CC(NC(=O)CC3COCC4(CCC4)O3)C2)=O)cc2cc(Cl)ccc2s1 c1(C(=O)NC2CC(CNC(=O)C(O)Cn3cncn3)C2)[nH]c2ccccc2c1Cl C1(NC(C2CCC(F)CC2)=O)CC1C1CCCN(C(=O)CCn2cnnn2)C1 C1(N=c2nc[nH]s2)(C(=O)OC)CCN(C(=O)C2CSc3ccccc32)CC1 N1(C(Cc2[nH]c(=N)sc2)=O)CCC2CCN(C(=O)Cn3ccc([N+](=O)[O-])n3)CC12 C1(CC)CC(O)CCN1C(=O)CC1CC(F)CN1C(c1ccc(OC)nn1)=O Nc1cc(C(=O)NC2CCCCC2NC(=O)C(F)OC(F)(F)F)nc(O)c1 C1(OC)CC(CC(=O)NCC2CC2NC(C2(CF)CC2)=O)C1 C1(O)(C(C(=O)NCC(CSC)OC)F)CN(C(=O)CCN(C)CCO)C1 c1(CC)[nH]nc(C(N2CC3C(C2)N3C(c2cccc(C(F)(F)F)c2)=O)=O)c1F c1(CNC(C2CC3CC3N2C(c2cc(C(F)(F)F)ccn2)=O)=O)ncccc1F C1(C(N2C(CNC(=O)CCCc3cccs3)CC(OC)C2)=O)CC(C(C)C)=NO1 CC(C)C(C(=O)N(C)CCN(C(=O)C(C)Sc1ccccc1)C)NC(N)=O Cc1c(C(c2nnnn2C2CCCC2)Nc2ccc(OCF)cc2)ccnc1F c1(OC)ccc(OCC(=O)NCCNC(=O)CCCCOC)cc1 CCCCC(CC)C(=O)NC(C1(CNC(=O)CCSc2ccccn2)CC1)C C1(C(N(C)CC2CCN(C(CSCC#C)=O)CC2)=O)CC2CCCC2C1 c1(CC(C(N2CCC(C(N)=O)(OCC)CC2)=O)N)ccc2c(c1)CCO2 CC(C)(C)CCC(C(=O)O)NCCC1CC1Cc1ccccc1 C(=O)(CCCCN=[N+]=[N-])NC(CCCC)C(=O)NC1CCC(CO)C1 O=C(C1COc2ccccc21)NC1CCN(C(=O)CCCCCF)C12CCC2 C1(CNC(C2N(C(C(CCC)OC)=O)CC=C2)=O)CCCC12CCC2 CCC(CNC(=O)CC1CC(O)C1(C)C)(CC)NC(=O)C(C)Oc1ccccc1 N1(C(c2c(CC)non2)=O)C(CNC(c2cc(C(N)=O)on2)=O)CC2COCC12 N1(C(Cc2ccc(C)o2)=O)CCC2(CC1)CC2NC(C1CC(n2cnnc2)C1)=O Cc1cc(C)c(C2CCCN2C(=O)C(=O)N2CC(CCF)C2)c(C)c1 C=C(C)CN=C(NCC1CCCOC1)NCC(c1ccc(OC)cc1)OC c1(NC(C(=Cc2cscn2)C)=O)cccc(N2CCCC2)c1 c1(CC(C)C(=O)NC2CN(C(c3cnc(C4CC4)[nH]3)=O)CC2O)ccc(F)cc1 N1(C(C2C(C)OCCC2)=O)CC=C(CCNC(c2cn(C)c(=O)nc2O)=O)CC1 C1(C(=O)NCC#C)CC2(CCN1C(=O)C(C)N1CC(C)C1)CC2 c1(C(=O)NCC2CCCN2C(C2CCCSC2)=O)cc2occc2s1 C(=O)(C1c2ccccc2CN1C(=O)CSc1nc[nH]n1)Nc1cnn(C)c1Cl c1(CC(=O)NCC2(NC(C=C(C)Cl)=O)CC2)cc(C)cc(C)c1 N1(C(C(=O)NC(C(=O)OC)C)c2csnn2)CCCC2(C1)NC(=O)NC2=O N1(C(C)C)CCCC(C(=O)NCC2CCCCN2Cc2cnc[nH]2)C1 Cc1cccc(C(=O)NC2(CO)CCN(Cc3ccccc3)C2)c1CO C1(C(=O)NCCOC2CCN(C(c3cc(CC)nn3C)=O)C2)NC(=O)C2CCC12 Cc1[nH]c2ccc(C(N3CCN(C(=O)C=Cc4ccsc4)CC3)=O)cc2c1C C1(C(N2CCC(=CCNC(C3CC3F)=O)CC2)=O)CC2CCC(C1)C2F CN1CC(C(=O)NC2CCCC2NC(C2(c3ccnn3C)CC2)=O)NC1=O N1(C(CNC(CC)=O)=O)CCN(C(=O)C(C2CC2)OC)C(c2cccc(Cl)c2)C1 Cc1ccc(C(N2CCC(CO)C(NC(=O)CC(C)(C)F)C2)=O)cc1[N+](=O)[O-] C1(COCCN2C(C)COCC2)CCCN1N1CCN(CCO)CC1C N1(C(c2ccc(C(C)C)s2)=O)CCN(C(C2CC3(CCC3O)C2)=O)CC(C)C1 C1(C#N)(C(=O)NCC2(C)CCN(C(c3c[nH]nc3F)=O)C2)CC2(CCC2)C1 C1(O)(CC(C(=O)N(CC(C)CO)C)NC(C=C(CCC)C)=O)CCCCC1 C1=CC(=O)NCc2ccc1cc2.C(=O)(C(C)C(O)CC)N1CC(O)(CCC)C1 C(=O)(CCCn1cccn1)NC(CC)CNC(=O)C(C)n1cncn1 C(CCN=C(NCc1ccc(C(C)(F)F)cc1)NCC(F)F)c1n(C)nnn1 C(CN=c1[nH]c2ccccc2s1)NC(N(CC(C)C)CC1CCCC(C)C1)=O N1(C(c2c(CC)ocn2)=O)CCN(C(=O)Cc2ncoc2C)C(C2CCCC2)C1 N1(C(c2ncc(C)c(C)c2)=O)CC2(C1)CN(C(C1CCC(F)C1)=O)CC2CO C1(CC(F)F)C(=O)N(CCCSC)C(=O)C(=O)N1C.C1(C)CCCCC1.CNC C1(C(N2CCC(O)(CNC(C(CC)N(C)C)=O)C2)=O)CC(C)(C)C(C)(C)C1 C(=O)(C(C)CC(C)C(C)=O)NC1CC=C(C(=O)NC(C(CCC)O)CO)C1 c1(C(=O)NCCNC(C2N(C)C(=O)NC2)=O)cnc2ccc(F)cn12 c1(C(N2C(CNC(C(C)SC(C)C)=O)CC(O)C2)=O)csc2c1CCCC2 N1(C(c2n[nH]c(C)c2Cl)=O)CCC2CN(C(C3CCCN3N=O)=O)CC2C1 Cc1cc(O)cc(O)c1C(=O)NCC12CC1CN(c1cc(N(C)C)ncn1)C2 C(=O)(C1CCCn2ncnc21)Nc1c2cnn(C(C)(C)C)c2ncn1 c1(OCC)cc(Cl)n[nH]c1=NCCN1CCC(OC)CC1 c1(CCNC(C(C)N(C(=O)C(C)NC(C)(C)CC)CC)=O)nccc(C)n1 c1(SC)ncc(C(N2CCCCC2CCCNC(=O)C=C(C)C2CC2)=O)c(O)n1 C#CCC(CC(=O)Nc1ccc(O)c(CO)c1)NC(=O)CC1CCC2CC12 CCCCCC(O)C(C)C(=O)NNc1cc(C(F)(F)F)n2ccnc2n1 N1(C(C(=O)NCCCF)CC2CCCC2)CCCCC1c1ncccn1 N1(C(C(CC)C)=O)CC(C2CCN(C(=O)Cc3ccc(CC(C)C)cc3)CC2)C1 N1(C(Cc2c(C)cco2)=O)CC(NC(=O)C(C)n2ccnn2)C(N=[N+]=[N-])C1 C12(CSC)CC(C(=O)NCC3(NC(=O)C(C)C#N)CCCC3)(CO1)C2 C1(NC(c2nc(C)oc2)=O)CC2CCC(C1)N2C(C1CCCC(C#N)C1)=O C1(C(N2CCC(N3CCN(C(C4(O)CC4)=O)CC3)C2)=O)CCCNS1(=O)=O CC(CC(=O)NC12CCC(CC1)CC2)C(C)(C)NC(c1cc2ccncc2[nH]1)=O N1(CCC)CCC=C(c2ccc3[nH]cc(CC(N4CCCCC4CO)=O)c3c2)C1 N1(C(c2cccc(C)c2Cl)=O)CC2=C(C1)CN(C(=O)CN1C(C)CCC1C)C2 S(=O)(=O)(c1csc2ccccc12)N1CCN(C(=O)Cc2ccc(O)cn2)C2C1C2 C1(C(N(CCNC(CSCC=C)=O)CCOCCC)=O)CN2CCCC1CC2 c1(SCCC(=O)NCC2(NC(C3COC(=O)C3)=O)CCOCC2)cccc(Cl)c1 C(C)(C(=O)NCC1CCCCN1C(c1n[nH]c(C)c1C)=O)(C(C)C)NC(C)=O N1(C(C(CC)C)=O)CCN(c2cc(OC(C)=O)ncn2)CC1c1ccccc1 c1(C(=O)NCC(C2CCCC2)NC(C(COC)(C)C)=O)cc(Cl)c(Cl)cc1C c1(C(=O)NCC(c2ccccc2)NC(C2CCC(=O)NC2)=O)ccc([N+](=O)[O-])[nH]1 C1(C(F)(F)F)(NC2CCC(CNC(=O)OC(C)(C)C)C2)CC=CCO1 CCCC(CNC(=O)C(O)CCN(C)C)C(=O)NCC1(F)CN(C)C1 C1(NC(C2C(=C)C2C(=O)OC)=O)C2CCC1CN(C(=O)C(C(C)C)OC)C2 c1(CC)cc(=NC(=O)C(CC(C)C)NC(=O)CSCC(F)F)[nH]n1C C1(C)(C(=O)NCC(CCCC)NC(=O)C(=O)C(F)(F)F)CCCS1(=O)=O c1(NC(C2(F)CCN(Cc3ccc(COC)o3)C2)=O)nc2cc(Cl)ccc2s1 C(CS(=O)(=O)CC(=O)NC1CN(C(=O)CC2COCCOC2)CC12CC2)OC C1(C(N(CC(C)OC)CC)=O)CC2(C1)CC(O)C2.C1(=O)CN1C.CC(C)C CC1CCN(C(=O)CCn2cccn2)CCN1C(=O)CCOCc1ccccc1 C1(O)(CCNC(c2ccc(CCC)[nH]2)=O)CCN(C(=O)CCc2ccsc2)CC1 c1(C(C(=O)N(CC(O)CNC(=O)CSCC2CCCO2)C)(F)F)ccc(F)cn1 C(CC(C)C)(C(=O)NCCCN(C)Cc1cn(-c2ccccc2F)nc1C)OC n1(C(C(N2C(CCNC(c3c(C)csc3)=O)CCC2)=O)C)c(C)cc(O)cc1=O C1(COC)CN(C(=O)CC2(C(F)(F)F)CCC2)CCN1C(c1ccccn1)=O N1(C(C(CC)(C)O)=O)CC(CNC(c2cc(Br)ccn2)=O)OC2(CCC2)C1 CN1CCCC(O)(CC(=O)NCC(C(C)(C)C)NC(c2ccncc2O)=O)C1 Cc1cnc(C(=O)NCC#CCNC(=O)Cc2cncc(Br)c2)c(F)c1 CCC(C)(C)C(=O)C(=O)N1CC(C(O)C(=O)NCCOC2CC2)C1 C(=O)(CC(C)CC(=O)OC)NCC(CC)N(C(=O)Cn1nnc(C)n1)C C1(C(=O)N(CCO)CCO)C2CCCC1CN(S(=O)(=O)c1nccs1)C2 N1(C(CC(C)CF)=O)CCN(C(c2ccccc2CN(C)C)=O)CC1C1CCC1 Cc1ccc2[nH]c3c(c2c1)CC(NC(C1C(CN)C1(C)C)=O)CC3 N1(C(c2c(C)cno2)=O)CCC2(CC1)CC2NC(c1nc(Cl)c(Cl)s1)=O C(CC(C)(C)CC(=O)N1CCC(CCC(=O)NC2COC3(CCC3)C2)CC1)OC C1(C(=O)NCC2(CN=c3nc(CC)[nH]s3)CC2)CCC2(CCCC2)C1 c1(C(=O)NC2CCC(CNC(CCN(C(C)=O)C)=O)C2)cccc2oc(=N)[nH]c12 c1(C(C)(C)C)cc(C(=O)NCCOC2CCN(C(C3(C#N)CCC3)=O)C2)on1 CCCCCCC(=O)NCC(=O)NCC(N1CCC(c2nncn2C)C1)=O N1(C(CC2CC(CN(C)C)C2)=O)CCN(C(=O)CCc2cncn2C)CC1 C1(F)(CNC(CN(C)C(=O)C2CC2)=O)CCCN(C(C2CCCCC(=O)N2)=O)C1 c1(OC)cnnc(C(=O)NC2CC(CNC(=O)CCOc3ccc(C)cc3)C2)c1 N1(C(C=Cc2cn(C)nn2)=O)CCC2(CCC2NC(C2COCC2(C)C)=O)CC1 CCC(C)(C(=O)NC1COC2(C1)CN(C(=O)CCNC(=O)OC)C2)C(N)=O c1(OCC)ccc(C(=O)NCCC2CCCN2C(=O)CC2(C(=O)OC)CC2)cc1 C1(C(=O)NCCCCNC(c2ccn(C)c(=O)c2)=O)CCCCC(F)(F)C1 C1(C(=O)NCC2C(CCC)CCC2)(C(=O)O)CCSCC1 CC(c1cccs1)=CC(=O)N(C1CCN(C(=O)C(=Cc2cccnc2)F)C1)C Cc1ccc(Br)c2nc(C(=O)NCC3(C(=O)O)CCCS3(=O)=O)sc12 N1(C(c2cnc(SC)nc2)=O)CC(NC(c2ncc(Br)cc2C)=O)C(C#N)C1 c1(C(N(C(c2ccccn2)C)C)=O)cc(F)cc(F)c1 c1(CCCC)cc(C(C(=O)NCC(=O)OCC)N(CC(C)(C)COC)C)n[nH]1 C1(NC(=O)NC2CCN(c3ccccc3)C2)CCC12CCCCC2 C(=O)(CC1=CCCCC1)NCC1(CNC(C2CCC(OC)CC2)=O)CC1 C1(OC)CC(NC(=O)CC(C)(C)C2CC2)CN(C(C2COC(=O)C2)=O)C1 c1(OCC(=O)NCC(N(C)C(C2CC3CC3C2)=O)C2CC2)ccc(F)cc1O N1(C(C=C(C)C)=O)CC2CC1C2NC(c1ccc(C2CCCCC2)o1)=O c1(C(=O)NCC2C3CN(C(C4(CCN(C)C)CC4)=O)CC32)cc2oc(Cl)cc2[nH]1 C12(CNC(C(COC)(C)C)=O)CN(C(=O)Cc3nn(C)cc3Cl)CC1CCO2 C1(C#N)(CN(C(c2csnc2C)C(=O)NC2(C)CC2)CC)CCOCC1 CCC(C)(CNC(C1(CCF)CC1)=O)NC(=O)C=CBr c1(CC(=O)NCC(CNC(CCC(=O)NCCC)=O)O)ccc(OCC)c(F)c1 CCCCC(CCCC)C(=O)NCC1C(C)CCN1C(c1ccc(F)c(Cl)c1)=O CN1CC(NC(=O)C(C2CCN(C(=O)CC3CCSC3)C2)F)C2(CC2)C1=O N1(C(CCNC(=O)NC)=O)CCN(C(C2CCC(F)(F)C2)=O)CC1CC(F)(F)F c1(-c2c(OC)snn2)nc(C(C)(C)C)nn1Cc1ccc(Br)cc1 N1(C(C)C)CCC(C(=O)NC2CCC(N(C)C(c3cnn(C4CC4)c3)=O)C2)CC1 CCCCCC(O)C(=O)N(C1CCCC1)CCCNC(=O)CCCC(C)=O N1(C(Cn2cc(C)c(O)nc2=O)=O)CCN(C(=O)CC2CC(=O)C2)C(C)CC1C c1(-n2cc(C(=O)NC(CCOC)CNC(C3CC(C)C3)=O)nn2)cccc(C)c1 C(CC(C(=O)N1CCC(SC)C1)NC(=O)CCc1cnccn1)OC C(=O)(C(CC(C)CC)NC(=O)CC=C(Cl)Cl)NC1C(C#C)CCC1 C1(C(=O)NC(CNC(c2cnc(CCCC)s2)=O)CO)CCc2nccn2C1 c1(CNC(C(CCOCC)NC(=O)CCc2ccccn2)=O)cc(C)cc(F)c1 CCC1CCCc2sc(NC(=O)CN(C)C(c3cn4c(n3)CNCC4)=O)nc21 C1(C(=O)NCCCNC(c2cnn[nH]2)=O)(CO)CC12CCC2 C1(C(N(CC(CC)NC(C(C)=CC)=O)C)=O)CCCCN1S(=O)(=O)CCCC C(=O)(CCCC(C)(C)C)NCCC(CC)(CC)NC(=O)Cn1ccc(Br)n1 C(=O)(CC(CNC(c1cc(C)sc1C)=O)C1CCC1)N(C(C(CC)C)C)C1CC1 c1(NC(N2C(CCNC(=O)OC(C)(C)C)CCC2)=O)cc(O)c2ccoc2c1 N1(C(COc2cc(C)on2)=O)CC2CCC1CN2C(C1(C#N)CC1C(F)(F)F)=O c1(C(N2CC(C)C(NC(C3(F)CCCC3)=O)C2)=O)[nH]cc2c1CCS2(=O)=O c1(Cc2nc(C3Cn4c(nc(C)n4)C3)on2)ccc2c(O)n[nH]c2c1 C1(OC)CC(C(=O)N(CC(N2CCCC2)C)C)N(C(=O)CCc2ccn(C)c2)C1 Cc1cc(C)c2c(c1)C(C(=O)NC1CCC(NC(=O)CCC(C)(C)C)C1)CCC2 N1(C(CCC(=C)C)=O)CC2CC1CC2NC(c1ccc2c(c1)CC2)=O N1(C(CC=CC=C)=O)Cc2ccccc2CC1CNC(C1OCCC1C)=O N1(C(c2ccc(OC)c(Cl)n2)=O)CC2(CCN(C(=O)CCC3CCCCO3)C2)C1 C#CCCCC(C)C(=O)N1CCCC1C(=O)NCC1CC2CCC2C1 C=CCC(CC=C)C(=O)N1CCN(C(C2CCCCN2CC)=O)CC1CF c1(C(=O)NCCC2CCC(NC(c3ccc(OC)cc3)=O)C2)ncnc(O)c1F CCC(C)CC(CO)N(C(=O)C(=CC1CCCC1)C)C1CCN1C(=O)CC(Cl)Cl C1(C(N(CCCN(C(=O)C(O)Cc2cn(C)cn2)C)C)=O)CCS(=O)(=O)C1(C)C Cc1cc(C#N)cnc1C(=O)NC1(C(=O)NC(CF)C(F)(F)F)CC(F)C1 c1(COC)nc(NCc2cnn(Cc3ccccc3)c2)cc(=NC(C)CSC)[nH]1 Cc1c(Cl)sc(Cl)c1C(=O)NC(C)CN(C)C(C1CC1c1nccn1C)=O CCN=c1[nH]cc(C(N2CC(NC(C3(C)CCCO3)=O)CC2C)=O)s1 C12(CNC(=O)C(F)CC3CCC3)CCC(NC(c3cc(Cl)cnc3O)=O)(CO1)C2 c1(C(=O)NCCC2(CNC(c3nc(OCC)oc3)=O)CC2)ccc([N+](=O)[O-])s1 C(C(CNC(C1CC12CCCCC2)=O)S(C)(=O)=O)NC(C1C(CC(C)C)C1)=O CCC(CC)(CCNC(c1nc(C)ccc1OC)=O)NC(c1sc(C)nc1C)=O C1(CNC(C2CCC(C)O2)=O)C(C2CC2)CCN1C(C1CCCCC1O)=O C1(C(=O)NCc2ccn(C)n2)CN(Cc2ccc(Cl)cc2O)CC(F)(F)C1 C1(NS(CC(OC)OC)(=O)=O)CC2(CO1)CN(C(=O)OC(C)(C)C)C2 CC(C)CCC(=O)C(=O)NC(CCC1CC1)C(=O)N(CCC(O)CO)C c1(CNC(C(C)N2CCCC2)=O)cc(C(=O)NC2(CC3CCC3)CC2)no1 C(=O)(CCCC1CCC1)N(C1CCCC1)CCNC(C(C1CCC1)OCC)=O C12C3CC4C1C4C3C(=O)N2.N1(C(CCNC(=O)OC)=O)CC(F)(C(=O)OC)C1 c1(CC(N2CCC(C(=O)Nc3cc(O)ccn3)C2)=O)ccc2c(c1)OCO2 N1(C(CCC(C)OCC)=O)CCN(C(C2CC(=C(F)F)C2)=O)CC(O)C1 N1(C(C(CSC)OC)=O)CCN(C(C2(OC)CCC(C)(C)C2)=O)CC12CCC2 c1(OC)c(CC(=O)NCC2C3CCC(C3)N2C(=O)C(O)C2CCC2)cccc1F c1(N(C)C2CC2)[nH]c(=NCC(F)(F)c2ccc(F)cc2)nc2scnc12 c1(C2CN(C(C)=O)C2)c(C(=O)OC(C)C)noc1C.C1(=O)C(CC2CCOC2)N1 C12(C(=O)NC(CNC(CCOCC#C)=O)(CC)CC)CC(CO)(C1)OC2C C(CCC(C)C)(c1n(C(CC)C)nnn1)NCCCNC(=O)OC(C)(C)C C1(COC)CC(N=c2[nH]c(=NCCCc3cnn[nH]3)c3cccc(F)c3[nH]2)C1 c1(CC)c(C(=O)N(CCCCN(C(=O)C(N2C(C)CCC2C)C)C)C)ccn1C N1(Cc2[nH]cc(C#N)c2)CC2CC(NC(C3CN(CCCO)C3)=O)CC2C1 C1(NC(c2c(C)nn(C)c2)=O)CN(C(=O)C(c2ccncc2)C)CCC1CO Cc1nc(Cl)cc(Cl)c1C(=O)NC1CCCN(C(=O)CC2NC(=O)NC2=O)C1 c1(OC)ccc(Cl)c(C)c1C(=O)NCCCCN(C(=O)C1=CCCCC1)C c1(C(=O)NC2CCC(CC(=O)NCC3(CC)CC3)C2)ccc(C#N)[nH]1 c1(SC(C)Cc2ccc(Cl)s2)cccc(-c2noc(-c3ccon3)n2)c1 C(=O)(CCCCCn1cnnn1)N1CC(NC(CC2ON=C(C)C2)=O)C(C)C1 c1(C(=O)NCC2C(CNC(CC(=C)C)=O)C2)ccc(OCCN(C)C)cc1 C1(CN(c2occc2)C2CC2)CC2(CCOC2)CO1 c1(C(=O)NCCCNC(C2CCC(C(=O)OC)C2)=O)c(C)oc(C)c1Br C12(NC(C=C(C)C(C)C)=O)CCC1CN(C(=O)Cn1ncc(Cl)c1C)C2 C1(NC(=O)NCC(c2ccccn2)C)CCN(C)CC1c1cnn(C)c1 N1(C(C(C2CCOC2)OCC)=O)CCC2CCN(c3cc(Cl)nc(C)n3)CC2C1 N1(C(CC(=O)OCC)=O)CC2CC2(CNC(=O)CC(C)F)C1 N1(C(CCc2cnc(C)s2)=O)CC(CNC(=O)CCc2cn(C)nn2)CC1(C)C c1(C(N2CC3C(NC(CC(=O)OCC)=O)(C3)C2)=O)ccc2ccccc2c1 c1(OC)ccc2oc(C(N3CC(NC(=O)C(CCSC)N(C)C)C3)=O)c(C)c2c1 N1(C(c2cnn(CC(F)(F)F)c2C)C(=O)NCCOC)CCC2CCC(C2)C1 C1(CCC#C)CCCN(C(C2(CNC(c3oc(CO)cc3C)=O)CC(=C)C2)=O)C1 Cc1cnn(C)c1C(=O)NCC(C)(CO)NC(=O)CCC(=O)c1ccc(Cl)s1 C12(C(N3CC(C)C(NC(=O)CN4CCCNC4=O)CC3)=O)CCC(F)(CC1)CC2 S(=O)(=O)(C(C(C)C)c1ccccc1)NCCCCC(=O)OCC C12(NC(C3C(CCC)CCC3)=O)CCC(NC(=O)CCOC3CCCC3)(CC1)C2 C(=O)(C1=NNC(=O)C1)N(C)Cc1cccc(CNC(C2C(OC)C2)=O)c1 C1(CC)(CC)CC(NC(c2cccc(O)n2)=O)CN1C(c1cnc[nH]1)=O CC(C)C(O)(C(=O)NCC(C(C)(C)C)NC(=O)Cn1cccn1)C(F)(F)F C1(NC(CN(C)C(N)=O)=O)CC(C2CCN(C(c3ccc(N)c(F)c3)=O)C2)C1 C1(C(C)NC(CCN(CCCCC)C)=O)CCN(C(C2CC2CC)=O)CC1 C(C(C)C)(C(O)C(=O)NCCc1ocnc1CNC(=O)CC(C)SC)OC c1(C(=O)NC(C(=O)NCC)(C)C)cnc(CNC(C2C=CCCC2)=O)nc1 c1(CN2CC3C(C(N(CCO)CC)=O)(C3)C2)ccc2cnn(C)c2c1 C(c1ccc(F)cc1Cl)=CC(N1CC(NC(C2(C)CC2(F)F)=O)C1)=O O=C(CC(C(F)(F)F)NC(C1CCCSC1)=O)NC1(C2CC2)CCOCC1 c1(C(=O)NCCCNc2ccc(F)cc2F)ccc2ncsc2c1 C1(OCCOCCNC(C2(C#C)CC2)=O)CCN(C(=O)CC2(OC)CC2)C1 N1(C(C2(C)CCC(C)C2)=O)CC2(C1)CN(C(c1cscc1F)=O)CCO2 Cc1cc(C(N2CC(NC(c3c(O)cccc3F)=O)C(O)C2)=O)ncc1Br C=CCC(C)(CC)C(=O)N1CC2(CC(CC#N)C2)C1 Cn1ncc(CCC(=O)NCCC2CCN(C(C3(O)CCC3)=O)C2)n1 c1(C(=O)NCCC2(CNC(CC3C(C)=NNC3=O)=O)CC2)noc2ccccc12 c1(C(=O)NC(CC)CNC(c2ccn(C)c2)=O)ccccc1OCC(N)=O C12(C(N3C(C)CN(C(c4nncs4)=O)CC3)=O)CCCCC1OCC2 C(=O)(C1=Cc2ccccc2OC1)NCC1CCN(c2c(C)c(Cl)ncn2)CC1C CCCCCCCC(=O)NCC1(C(=O)NC(CO)CC(F)(F)F)CCC1 C1(NC(C(CC)C(C)C)=O)CC2(CCCN(C(c3coc4c3COC4)=O)C2)C1 N1(C(CCC#C)=O)CC(F)(F)CC1(C)CNC(=O)CC(C)P(C)(C)=O c1(CSCC(C)C)ccc(C(=O)NC2CCCC2NC(c2cnsn2)=O)o1 CC(CCCCCO)NC(C1CCCCC1CNC(=O)CC1OCCC1(C)C)=O C1(C(=O)NCCN(CCCCCC)C(c2cnns2)=O)CCCC(C(N)=O)C1 C1(C(=O)OC)(CNCC2(C(=O)NCC(C)(C)C(=O)NC)CC2)CCCCO1 N1(C(C(CCC)NC(c2ccc3cccnn23)=O)=O)CCc2n[nH]cc2C1 N1(C(c2ccn(CC#N)n2)=O)CC2CCC(NC(=O)C=CCF)(C2)C1 c1(C(=O)NC2CC(C)(CNC(C(C)n3ccnn3)=O)C2)ccnc(C(=O)OC)c1 CC1CCCN(C(c2cnn(CCF)c2)=O)C1CNC(=O)CN1CCC(O)CC1 C(C(C)(C(=O)NCCCC(=O)NCCC1(O)CCOC1)OC)OC C1(C(C2(C(N(CC)Cc3ccccc3)=O)CC2)=O)CCN(C(C2CC2F)=O)CC1 C12(NC(CCCCSC)=O)CCCCCC1N(C(=O)CCc1cn(C)nn1)CC2 c1(CC(=O)OC)c(C(c2ccc(N3CCCCC3)nc2)=O)[nH]c(C)c1C(=O)OC Cc1cc(C(N2CCC(F)(C(=O)NCc3c(F)cccc3F)C2)=O)cc(C)c1O c1(CCNC(C(C2CCN(Cc3ncnn3C)CC2)C)=O)cccc(Br)c1 C(=O)(CS(=O)(=O)CC)N(CCNC(c1nc(COCC)sc1)=O)C1CC1 c1(C(=O)NC2CC3(CN(C(C4CN(CC(C)C)C4)=O)C3)C2)ccc(N)c(Cl)c1O Cc1nc(O)nc(O)c1CC(=O)NC1CC(F)(F)CC1NC(C1CC=CCC1)=O CC(C)C(C)(CNC(=O)C(=O)NC1CC1)NC(=O)CC1CC2CCC1C2 C1(C(=O)NCC(CC)(C)Cl)CN(C(c2cc(C#N)cs2)=O)CCN1C C1(OC)CC(OC(C)(C)C)CN(CC2CNC(=O)C2)C1 C1(NC(C(C)NC(C)(C)C)=O)CN(C(C2CC3C=CC2CC3)=O)CCC1C C(=O)(C(CNC(c1nc(O)sc1C)=O)CC1CC1)NC(c1nc(C)[nH]n1)C C1(C(N(C2CCCOC2)CC)=O)CC2CCC1N2C(C1C2CC(=O)CC12)=O O=C1CCN(C(=O)Cc2ccn(-c3ccccc3)n2)C(C2CC2)C1 C1(NC(c2c(C)cc(F)s2)=O)CCC2(CCN(C(C3(N=[N+]=[N-])CC3)=O)CC2)C1 C1(NC(COC)=O)CC12CC(NC(C1(CO)CCCCO1)=O)C2 Cc1ccc(C=CC(=O)NCc2cc(C(=O)NCC(O)(CO)CO)no2)cc1 C(CNC(=O)CCc1cn[nH]c1)(C(=O)NC(C)(CO)C1CCC1)N(C)C C1(CNC(C(C2CC2)OC)=O)CN(C(c2cccc(F)c2)=O)CC1C(F)(F)F N1(C(C(C)OCCOC)=O)CCC(C)CC1CNC(=O)C(C(C)C)NS(C)(=O)=O c1(OCC(=O)NC2CCCC(NC(CCSCCOC)=O)C2)cc(F)cc(F)c1 C1(C(C)C)CCCC1C(N1CCCC1CNC(=O)CCc1ccccn1)=O C1(C(=O)NC(C)(CC)CC)(CC)CCN(C(c2nccn2C)=O)C1 C1(C(=O)NCCc2c(CNC(C(CC)F)=O)nco2)CC12CCCCCC2 C1(NC(c2nnc(C)s2)=O)CCN(C(C2(CO)CC(F)(F)C2)=O)CC1(C)C C=CCC(CC=C)C(=O)N1CCC1(C)CC(=O)NC(c1ncc(C)[nH]1)CC c1(C(N2CC(CNC(c3cc(OC)ncn3)=O)C2)=O)cc(F)cc(F)c1O C(c1ccncc1)=CC(=O)NC1(C(=O)NC(c2nc(C)sc2)C)CSC1 S(=O)(=O)(C=Cc1ccccc1)N1CCN(CC2(C)CCCN2)CC1 C1(C(=O)NC2(CCCC)CC2)COCCC1NC(c1occc1COC)=O c1(C(N(CCC(=O)NCC2N(C)CC(O)C2)CCCO)=O)ccc2cc[nH]c2c1 c1(C(N2CC(NC(C3CCCN(C)C3)=O)C(O)C2)=O)cccc2nccnc12 c1(C(=O)NC2C(CNC(C(c3cscn3)N(C)C)=O)CCC2)ccc2c(c1)CC2 CC1CN(C(=O)Cc2cccc(C3CC3)c2)CCN1C(C1CCCN1C)=O c1(C(N2CC(NC(CCC3CC(OC)C3)=O)C2)=O)nn(C)c2ccc(F)cc12 CC(CCNC(C1CCCCN(C(=O)Cc2cnns2)C1)=O)C(C)(C)C N1(C(=O)CC2CC2)CC2CC(C1)CN(C(C1CCC=CCCC1)=O)C2 N1(C(c2c(CNC(=O)C=Cc3cncs3)ocn2)=O)CCC(O)CC1C1CC1 N1(C(c2c(C)cco2)=O)CCC(NC(=O)CC2CCCCCCC2)CC1C c1(-n2c(-c3ccc(-c4ccc(I)c(F)c4)cc3)nc(C)n2)cccc(C#N)c1 c1(C(=O)NC2CC(CNC(c3ccoc3Cl)=O)C2)ccc2cnccc2c1 c1(OC)ccc2c(c1)CC(C(c1nnnn1C)Nc1ccc3nc(C)sc3c1)CC2 Cc1ccc(C(=O)NCC2CN(C(=O)C(c3ccc(C)s3)C)CCC2C)c(C)c1 c1(SC)cccc(C)c1C(=O)NC1CC1NC(=O)CCc1c(Cl)cccc1Cl C1(C(C)C)CCC(C)CC1C(=O)NCC(CNC(=O)CN(C1CCC1)C)CO C=C=CCN=c1[nH]c2c(c(=NCC3(C)CCOCC3)[nH]1)CCCC2 C12(CC(O)C1)C(=O)N2.c1(C(N2CC(C(C(=O)OC)O)C2)=O)[nH]ccc1C C12CC3(CCCN3C1=O)C2.N1(N(C(=O)C(C)C)CC)CC(C(=O)OC(C)(C)C)C1 C(c1cccc([N+](=O)[O-])c1)=CC(N1CCN(C(C(CCCC)C)=O)CC1C)=O C1(F)(C(=O)NCCSCC)CCN(Cc2cscc2Br)C1 C1(F)(C(=O)NC2CN(C(C=C(C)c3ccco3)=O)CC2F)CC2(CCC2)C1 CCCC(C#N)C(=O)NC(C1CC1C(N1CCC2CCC12)=O)C N1C(=NCCC(=O)N(C)C)NC1C.C12(CC(C)(C)C)CCCC1CC(=O)N2 C1(C2CCCCC2)(NC(C2(F)CCN(C(C3CCC(=O)C3)=O)C2)=O)CC1 c1(CNC(C(c2ccccc2Cl)NC)=O)ccc(OC(F)F)c(C)c1 c1(C(C2C3COCC23)NCC2(CCOCC)CCC2)nnnn1C1CCC1 c1(OCCC(=O)NC(C)CCCNC(=O)CC2CCCC2)ccccc1F C(=O)(C1=CCS(=O)(=O)C1)NC1CC(NC(c2ccc(N)cc2F)=O)C12CCC2 c1(C(N2CCC(NC(C(C(C)C)n3cnnn3)=O)C2)=O)ccc2ncccn12 CCC(C)C(C)C(=O)NCCSCC(=O)NCCCn1ccnn1 C1(NC(C(CCC)F)=O)CC(NC(c2ncnn2CC)=O)C12CCC2 c1(C(N2CC(NC(C3(OCC)CCSCC3)=O)C(C)C2)=O)ncn2c1CCC2 C1(NCC)CCN(C(C2CC3CC3C2)=O)C1 C(=O)(C(C)=Cn1ccnn1)N1CC(C)CC(CNC(CCSC)=O)C1 C12(NC(C3CC(OCC)C3)=O)CCCC(NC(=O)CCn3ccnn3)(C1)C2 C1(C)(C(=O)NCCCN(C(=O)Cc2csc(Cl)c2)C)CCNC(=O)C1 C1(CC(=O)NCC(CNC(C2(F)CC3(CCC3)C2)=O)CO)CC(=O)NC(=O)C1 N1(C(CCCSC)=O)CCC(CCCCNC(C2CCOC2C(C)C)=O)CC1 c1(C(=O)NC(C(C)NC(=O)C=CS(C)=O)CO)ccc(C(C)(C)C)c([N+](=O)[O-])c1 N(C(=NCCCCOc1ccccc1)NC1CC1)Cc1c(C)noc1C C=CCCCC(C)(C)C(=O)NC1CCCCC1CC(=O)NC1CCC12CCCC2 c1(C(=O)NC2CCCN(C(CN3CC(C)C3)=O)CC2)cc(F)c2c(c1)CCC2 N1(C(C23C(CN(C(CC4CCC(=O)CC4)=O)C2)C3)=O)CCC2(CCC2)C(O)C1 C(C(CC(C)C)C(=O)NC1(C(C)(F)F)CC1)NC(C(C)=CC(C)(C)C)=O c1(C(N2C(CNC(C3COCC3C(F)F)=O)CC(OC)C2)=O)cn(C)c(=O)n1C N1(C(=O)Oc2ccc(F)cc2)CC2CCC(F)(F)C2C1 c1(C(=O)NC2(CCC(=O)NC3CCN(C(C)=O)CC3)CCC2)ccc2cncn2c1 c1(NC(C2(c3ccc(Cl)cc3)CCC2)C)nccc(F)n1 C12(C(N3C(C(N(C)CC4(C)CC4)=O)CC(O)C3)=O)CC(C)(CCO1)C2 c1(C(=O)NC2C3OCC(NC(COCC#C)=O)(C3)C2)ccc2c(c1)C=CCC2 c1(C(=O)NC(CN(C(=O)CCOC)CC)C)nsnc1O CC(=Cn1ccnn1)C(=O)N(CC(C)CNC(=O)CCCn1ccnc1)C CC1CC(NC(c2cnc(O)c(Cl)c2)=O)CN(C(c2ccco2)=O)C1 C1(NC(c2nc(OCC)oc2)=O)CCN(C(c2cncc(Cl)c2)=O)CC1(C)C C(CC(=O)N1CCOCC(CO)C1)(C(F)F)NC(c1n(CCC)ccc1)=O C1(C(=O)NCC2CN(C(=O)CC(F)F)CC23CC3)(OC)CCS(=O)(=O)C1 CC(CC1CC(F)(F)C1)C(C(=O)NCCC1CC1)N(C1CCN(C)C(=O)C1)C C1(CCCNC(C(CC(=C)C)OC)=O)CCN(C(=O)CCOC(C)C)CC1(F)F C1(CN(C(C2(C)C(C)C2)=O)C)CCCN(C(=O)C(C)(C)CC2CCC2)C1 N1(C(c2c(C)cc(C)s2)=O)CCC2CN(C(c3ncc(F)cc3F)=O)CCC2C1 c1(C(=O)NC(C2CCCCC2)CNC(=O)CCC(F)(F)F)cccn2cnnc12 N1(C(C2CC(C)NC(=O)C2)=O)CCC2(CCC(NC(=O)C3=NOC(C)(C)C3)C2)C1 CC1(C(=O)NC2CC(F)CN(C(c3cccc(Cl)c3)=O)C2)CC(C(F)(F)F)=NO1 N1(C(CN(C)C2CC2)=O)C2CCC1CC(NC(C1CC(=O)N(C)C(=O)N1)=O)C2 C1(CNC(c2c(C)n[nH]c2)=O)CCC(CNC(C2CCCCC2C)=O)CC1 N(C1CCc2cccnc21)C(C1C(C)(C)CCN(C(=O)C2=NOCC2)C1)=O C1(C(N(C(C)CN(C)C(c2cn(C(C)(C)C)nn2)=O)C)=O)COCCN1C c1(C(N(C2CCCN(C(C3(C)CC4CCC3O4)=O)CC2)C)=O)ccc(F)cc1Cl C=CCC(CC(C)C)C(=O)N1CC2(CCC(NC(=O)C(O)C(F)F)CC2)C1 C(=O)(C(C)CS(C)=O)N(C1CCC(CNC(c2c(C)n[nH]c2C)=O)CC1)C C12(CC(=O)NCC(C)CNC(=O)C=CCF)CC3CC(C1)CC(O)(C3)C2 c1(CCCSCC(=O)NC2C(NC(C3(C#N)CC3)=O)C2)ccccc1 Cc1cc(C(=O)NCC(C(N2CCN(C3CC3)C(=O)C2)=O)N(C)C)cnc1C CCC(O)C(C)C(=O)N1CCCC(CNC(=O)CC2CCC2)C1 c1(C(=O)NC(C)CCNC(C2(C(N)=O)CCC2)=O)cc2c(Br)coc2cn1 CC1CCCC(C(=O)NC2CC(CNC(C3(CC(F)F)CCC3)=O)C2)CC1 N1(CCC(=O)N(C(C)C)CCNC(=O)CC2CC(=O)C2)CCCCC1C CCC(C)(C(=O)N1CCCC(NC(c2ccnn2CC#N)=O)C1)C(N)=O C=CCCC(C1CC1)NC(=O)CN(C(=O)COC1CC(NC(=O)C(C)C)C1)C c1(CNC(C(N2CCCCC2)C)=O)ccc(CNC(C2OCCC2C)=O)cc1 C1(CC=C)(N(C(=O)CC(O)CC)C2CC2)CCN(C(c2nc(C)oc2C)=O)C1 N1(C(c2oncc2C2CC2)=O)CCC(O)(CNC(C2(CF)CC2(F)F)=O)C1 c1(CC)ccc(-n2cnc(C(=O)NCC(O)CCNC(=O)C(C)OC)c2)cc1 c1(C(N2CC(CNC(COCCC)=O)C3C2C3)=O)cc(OC)cc(F)c1 n1(CC)ncc(C(=O)NCC(C(C)C)NC(C2(C)CC=CCC2)=O)c1Br c1(CC2CCCO2)ncc(CNC(=NC)NN(c2ccccc2)C)s1.CC C#CCC(CC(=O)NC(c1snnc1C)C)NC(=O)C(C)(C)COC Cc1ccc(N(CCO)C(=O)NCc2ccnn2C2COC2)cc1 N1(C(C(C)OCC)=O)CCN(C(=O)C(C(C)C)NC=O)CC(O)C1 C12(CNC(=O)CSc3ccc(F)cc3)CC(CC1C(=O)O)C2 Cc1cc(CNC(C2(C)CCN(C(=O)CCC(C)(F)F)C2)=O)cnc1F c1(C(C(=O)OC(C)(C)C)N(C(C(CC)C2CCC(=O)N2)=O)C)ccc(SC)cc1 N1(C(C2C(C(C)C)C2)=O)CC2CC(NC(c3cnn4cccnc34)=O)CC1C2 C1(C)(C(N(CC(C)N(C(CC2(COC)CC2)=O)C)C)=O)COCCO1 C(=O)(C(C(C)(C)C)C1CCCC1)N1CC(O)(CN(C(=O)CC2CCOC2)C)C1 c1(OCC)cc(N2CC(NC(=O)C(c3ccc(OC)cc3)=O)CC2C)nc(C)n1 C1(C(N(CCC)C(C)C)=O)COC2(CCN(C(=O)CS(=O)(=O)CC)CC2)C1 Cc1cc(C(=O)NC2CCC(C)N(C(=O)CCOC3CCCC3)C2)c(N)c(Cl)c1 N1(C(CC2(C)CC2(F)F)=O)CC2CC2(CNC(C2(C3CCC3)CC2)=O)C1 c1(C(=O)NC(C(C)NC(C=CC(C)C)=O)(C)C)ccc(C#N)n1C CCCCCC(C)CC(=O)N1CCC(N(C(C2CC(CCO)C2)=O)CC)CC1 N1(C(C(C)OCC(F)(F)F)=O)CCOC(CN(C(=O)C(=O)NCC2CC2)C)C1 c1(N2CC(COC)OCC2)cc(Br)ccc1S(=O)(=O)N1CC2CC1CS2 c1(OC(C)C(=O)NCC23CC(CN2C(c2ccoc2)=O)C3)ccc(Cl)cc1 N1(C(C)=O)CCOC(C(N2CCCC2C2(NC(C3CC=CCO3)=O)CC2)=O)C1 N1(C(C2C(C)OCCO2)=O)CCC(C(=O)NCCC(C)(O)C2CC2)CC1C N1(C(C(c2ccc(F)cc2)C)=O)CC2CCN(C(c3cnc(Cl)[nH]3)=O)C2C1 Cc1cc(C(=O)NC2C=CCN(C(=O)C(C)CO)C2)nn1-c1ccccn1 Cc1nc(C(N2CC(CC(=O)N(C34CC(C3)C4)C)C(C)C2)=O)cn1C C=CCN=C(NCc1ccsc1C(F)(F)F)NCC(C1CCOC1)OCC C1(NC(=O)C=C(Cl)Cl)(CO)CCCN(C(=O)C(O)C(F)(F)F)C1 c1(C(=O)NC(C2CCN(C(c3cc(COC)sc3)=O)C2)C)nnn(C)c1C(F)F Cc1ccc(C(=O)O)cc1.c12ncnc(n1)CC(=O)NN(C)CC1CCN2C1 c1(C(=O)NC2CC(CNC(c3c(OC)ncc(F)c3)=O)C2)cccc2ncnn12 O=C(C1=C(Cl)CCOC1)NCCC(O)CNC(C1(CC(F)F)CC1)=O c1(C(=O)NC(c2cn(CCCO)nn2)C)nn(C)c2c1CCCC2 c1(C(=O)OCC(C2(CS(C)(=O)=O)COC2)=O)nc(Cl)cs1 C1(CNC(c2ccn(CCC)n2)=O)CN(C)CCN1C(C12CSCC1C2)=O Cc1onc(C(=O)NCC(CNC(c2c[nH]c3ncccc23)=O)CO)c1[N+](=O)[O-] C(N=c1[nH]c(=NCC2OCc3ccccc32)[nH]c2c1CSC2)C1C(C)CCC1 CC(C)C(N=[N+]=[N-])C(=O)NC(CCN(C)C)C(=O)N(CCS(N)(=O)=O)C C(C)(CCCCNC(c1ccc(C(C)(F)F)cn1)=O)NC(C(C)OCC(C)C)=O C(CC(O)CC(=O)N1CCC(CC(C)NC(=O)Cc2csnc2C)CC1)SC Cc1cc(C(C)C)nc(=NCCCCNC(=O)Cc2cc(C3CC3)on2)[nH]1 C1(CNC(C2CC(=O)N(O)C2)=O)CC12CCN(C(=O)CCOCC1CCC1)CC2 c1(C(=O)NC2CN(C(c3ccco3)=O)CC23CC3)cc(Br)ncc1Br C(C)(C(CC(=O)NCC(O)(C1CC1)C1CC1)NC(c1c[n+]([O-])c(C)cn1)=O)OC C1(CCCNC(C=CC=CC)=O)CN(C(C23CC(OC)(C2)C3)=O)CCO1 C1(N(C)C)(CC)CCCN(CC(=O)Nc2cccc(C#N)c2)C1 N1(C(C(C)(C)C#N)=O)CC2CCC(NC(=O)CC3(O)CCOC3)CC2C1 N1(C(CC(CC)C)=O)CCC(C(N2CCC(NC(=O)NC)C2)=O)C(C)(C)C1 c1(NC(C2(F)CCN(Cc3ccc(F)cc3)C2)=O)ccc(F)c(CO)c1 C=CCC(CC=C)C(=O)NCC1CCN(C(C2CCC2(C)C)=O)CC1C NC(=O)CCCCC(=O)N1CC(CNC(=O)CCC2CC2)OC(C(F)(F)F)C1 C1(CNC(=O)Cn2nnc(=O)[nH]2)CCN(C(=O)CCc2cnc[nH]2)CC1(F)F C(CCC(=O)N1CC(C)(CCC(=O)NCC2CNC(=O)C2)C1)OCC Cc1ncccc1CC(=O)NCCC(O)CNC(c1ccns1)=O CC1CC2(C1)CC(N=c1nc(N3CC4CC3CS4=O)c3c([nH]1)CSC3)C2 N1(C(C2CN(C)CC(C)O2)=O)C2CCC(C(=O)NC3CCCCCC3F)C1CC2 N1(C(CSCC#C)=O)CCC(F)(C(=O)NCCC2CCC(C)O2)CC1 Cc1cc(-c2ccc(C(=O)Nc3ccno3)nc2C)cc(C)c1 C#CC1(C(=O)NC2CCCC2NC(=O)CCc2ccc(Cl)nc2)CCOCC1 CS(=O)c1cccc(NC(c2nc(Cl)sc2Cl)c2nnnn2-c2ccccc2)c1 S1(=O)(=O)c2cccnc2N1.Cc1nc(C(C)C)ccc1CNNC1COC(C)(C)C1 c1(C(=O)NCCCCN(C(CCN(CC(C(C)C)C)C)=O)C)occ2c1CCC2 Nc1cc(C(=O)NCC(CO)NC(=O)CCc2ccoc2)ccc1Br c1(-c2cn(C(C)C(C(=O)CCCC3CCCC(=O)N3)=O)nn2)cc(C#N)ccn1 c1(OC)cc(F)c(C(N2CCC3(C2)CN(C(=O)CSCCN(C)C)C3)=O)c(Cl)c1 C1(C(=O)NCC23CC(NC(=O)CS(=O)(=O)N4CCCC4)(C2)C3)CC12CCSCC2 C1(NC(C(C)(C)SC)=O)CCN(C(c2ccc(C(C)=O)[nH]2)=O)CC(O)C1 c1(C(N(C(CNC(C(CC)O)=O)C)C)=O)cc(C(F)(F)F)c(C)c([N+](=O)[O-])c1 C12(C(=O)NC3CN(C(c4cccc5nc[nH]c45)=O)C3)CCCCC1CC(F)(F)C2 CCC(CNC(c1cc(CO)on1)=O)(CC)NC(=O)C(=O)NCCNC(C)=O c1(C(C)C)nc(NCCC2SCCS2)cc(=NC2CCCC(N(C)C)C2)[nH]1 c1(C(N2CC(C)(C)C(CNC(=O)CC3CC34CC4)C2)=O)ccc2c(c1)COCC2 CCCC(C)(CC)C(=O)N1CCN(CC2(NC(c3oncc3C)=O)CC2)CC1 CC1(C)CCCC(C(=O)NC(C)(CNC(c2c[nH]nc2F)=O)CO)C1 c1(C(N2CCC(CN(c3ncc(I)cn3)C)C2)=O)ccnc(Cl)c1F c1(C(=O)NCC2CC(CNC(C(CC)(F)F)=O)OC2)ccc(C=NOC)cc1 Cc1oc2ccccc2c1C(N1CCN(C(C2CCCC2CF)=O)CC1)=O Cc1nnc(CCC(=O)NCC(C2CC2)NC(=O)CC(=O)OC(C)(C)C)n1C c1(CC(=O)NC(C)CNC(=O)CN2CCCC2CO)cnn2ccccc12 N1(C(C2C3CCN(C(c4ccc(NC)cc4)=O)CC32)=O)CC2(C1)CC(C)(F)C2 CCCC(C)(C)NC(=O)NCc1ccc(-c2sccc2C)s1 Cc1nc(CC(=O)NC2CC(C(=O)NC(C3CCC3)C)C2)c(C)s1 C=CC1(CO)CCN(C(c2c(CNC(C3CC(O)C(F)C3)=O)cnn2C)=O)CC1 c1(NC(N2CCN(c3ncccn3)CC2)=O)ccc(C(N2CCCC2)=O)c(Cl)c1 c1(C(=O)NCC(COC)NC(c2cocn2)=O)cccc(N(C)C)c1 O=C1CCc2cc(S(=O)(=O)N3CCC4CCCOC4C3)cc3c2N1CC3 CCCC(CC)CCC(=O)NCCC(CNC(=O)Cc1cc(C2CC2)no1)OC C#Cc1ccc(C(N2CCC(N(C(=O)C(c3cnccn3)C)C)C2)=O)cc1 C1(NC(C=C(COC)C)=O)CCC(C)(CNC(=O)C(F)=C(C)C2CC2)C1 C(=O)(CC(O)C(C)CC)NC1CC(NC(c2cc(CCC)nc(O)c2)=O)C1 c1(CC)ccc(C(N2CC(NC(=O)COC3(C)CCCC3)CCC2C)=O)cc1F C1(C(N2CC(NC(C(C)CC3CCC3)=O)C(O)C2)=O)CCc2ccccc2CC1 c1(NC(c2n(CCC)nnn2)c2cn(C3CCC3)nn2)ccc(Cl)c(C(F)F)c1 C1(C(CNC(C2(SC)CC2)=O)=O)CCCC(O)C1.C(C(C)N(C)C=O)N C=CCCC(CC(C)C)C(=O)N1C(CNC(c2coc(SC)c2)=O)CC2COCC12 C1(CC(C)NC(C2CC(CF)C2)=O)CCN(C(=O)COC2CCCOC2)CC1 C1(CC(=O)NCC2(F)CN(C(C3(CN(C)C)CCCC3)=O)C2)CN2CCC1CC2 C#CC1(O)CCCN(C(=O)CC2(C)CCN2C(=O)Cn2nc(C)cc2C)C1 C1(NC(=O)Cn2cccn2)CN(C(C23CSC(C2)C3)=O)C2CCCCC12 c1(C(=O)NCC2C=CCN2C(c2cocn2)=O)ccc(OC(F)(F)F)cc1Cl N1(C(c2c(C)c[nH]n2)=O)CCC2(NC(c3[nH]nc([N+](=O)[O-])c3Cl)=O)CCCC12 C(CCCC(c1nnnn1-c1ccccc1Cl)NCC1(C)CCC(=O)N1C)(OC)OC O=C(C1=CC2CCC(C1)C2)NCc1cc[nH]c1C(=O)NCC1CCC(O)CC1 C1(NC)CCCN(C(=O)C(=O)NCC(c2ccco2)NCC)C1 N(C(=NCCc1cccs1)N1CC2C(C(F)F)C2C1)CC1(CF)CC1 N1(C(C(C=C)(C)CC)=O)CC2CCN(C(=O)CSc3n[nH]c(O)n3)CC2C1 CN1CCN(C(=O)C(CC(F)F)N(C(=O)CC2CC=CCC2)C)CC1=O N1(C(c2c(COC)noc2)=O)CCC2(CCN(C(=O)C(C)(O)COC)CC2)C1 C1(NC(C2(COC)CCOCC2)=O)CN(C(C2(C)CC2(F)F)=O)CCC1CO C1(C(=O)NC2CN(C(=O)C(F)CC3CCOC3)C2)OCC2CCCC1C2 c1(C(=O)NCC2(C)OCCN(C(Cc3cn(C)nn3)=O)C2)onc2ccccc12 C(C(C)(F)CNC(c1ccc(CO)s1)=O)NC(C=CCN(C)CC)=O n1(CC(N2CCCCC(NC(C(C)(C)C3CC3)=O)C2)=O)cnc2c(N)ncnc12 C1(OC)C(C)(C)CN(C(C2(C3CCCO3)CC2)=O)C1(C)C N1(C(C(CC)(C)OC)=O)CCC(NC(c2cnnc(C)c2)=O)CC(C)(C)C1 C1(CCC)(NC(=O)CN(S(=O)(=O)CC)C)CCCN(C(C2(C)CCNC2=O)=O)C1 CCC(C)(CNC(=O)C=CCOC)C(=O)NC1CCCCC1C N1(C(CCC#C)=O)CCC(C)C(NC(=O)CC(C)(C)c2ccccc2)C1 N1(C(CSCC(C)C)=O)CC2(CCN(C(C3CC3F)=O)CC2)CC1C C1(NC(CCS(=O)(=O)N(C)C)=O)CCCC12CN(C(C1(CCF)CC1)=O)C2 N1(C(Cn2c(CC)ncc2)=O)CCC2(NC(=O)C3=CCC3)CCCC12.C1(=O)CN1 c1(NCC2(N(C)C)CCC2)ccc(S(=O)(=O)NCC2(Cl)CC2(F)F)cc1Br N1(C(C2OCCC(C)(C)C2)=O)CCC(C(=O)NC2CC(OCCO)C2)CC1(C)C C1(C)(CNC(C(C)NC(C)=O)=O)CCCN(C(=O)CCS(N)(=O)=O)C1 C1(C(=O)OC)(C(C)C)CC1CNC(C)C(=O)NCC(F)(F)F CCC(CC)C(F)C(=O)N(C(C)CNC(=O)C(n1cc(C)cn1)C)CC N1(C(C(C(C(C)C)O)C)=O)CC(C(C)(C)C)Nc2ccccc21 Cc1ccccc1CC(=O)NCCC(C)NC(=O)C(=O)NCC1CC1 C1(CN(C(CCC#C)=O)C)CCCCN1C(c1cnc(S)[nH]1)=O C1(CC(=O)N(CC(CN(C(=O)CCS(C)=O)C)O)C)CCCCCCC1 N1(C(C2C(CC)OCC2)=O)CC(CNC(=O)C=CSCc2ccco2)CC(C)C1 N1(C(c2sccc2CO)=O)CCC(OCC(=O)N(CCO)C2CC2)C1 C1(CNC(c2c(CC)scc2)=O)CN(C(=O)C(C)SC)CCO1 CCS(=O)CC(=O)N1CCC(C)C1CNC(=O)Cn1ccnn1 c1(NC(C(=O)NCC2CCC=CCC2)=O)ccc(S(=O)(=O)CC2CCOC2)cc1 C=CCCC(O)CN(C)C(c1sccc1CNC(=O)CC1CC1(C)C)=O Cc1ccc(C(N2CC(NC(c3ncc(F)cc3F)=O)C(C)(C)C2)=O)cc1O C=C=C(C)CC(=O)N(C)CC1CCN(C(c2ccc(C3CCCO3)nn2)=O)C1 N1(C(C(C)Br)=O)CCCC2(CCCN2C(=O)C(C)Oc2ccccc2)C1 C=CC(CC)C(=O)NC1CCOC(CNC(=O)CCc2nccn2CC)C1 C(C(C)C(C)C(=O)N1CC2CC1(CNC(c1c(Cl)nsc1Cl)=O)C2)OC C(=O)(C1CCCc2cncn21)NC1(C2CCCN(C(C3CC(C)(O)C3)=O)C2)CC1 C(=O)(C(CCC(C)OC(C1CCOC(C(C)C)C1)=O)C(=O)OC)OC Cc1cc(F)ccc1NC(C1(C)CCN(C(C2CC2C(C)C)=O)CC1)=O N1(C(CC2CC(OCC)C2)=O)CC(O)CC1CNC(C1CC2C=CC1C2)=O Cc1cnn(C)c1C(=O)NCC1(O)CC(CNC(=O)CCS(C)=O)C1 c1(C(=O)NCC(=C)CCNC(=O)CCC2CCCC2)ccc(SCCCO)cc1 C1(C(N2C(CN(C(CCOC)=O)C)CCC2)=O)CCCCS1(=O)=O C1(CC)CN(C(=O)C(C)(C)C(C)C)CCN1C(c1nn(CC)nc1C)=O c1(C(N2CC(OC)C(NC(C34CC(F)(C3)C4)=O)C2)=O)cnc2n1CCC(C)C2 c1(C(=O)NC2CCC(NC(CN3CCC(C)C3)=O)CC2)ccc(F)c(C(F)F)c1 C1(C(F)(F)F)(NC(=O)NCC2(CC(C)C)CC2)CCc2ccccc21 c1(OC)ccc(C(N2CC(CNC(=O)Cc3ncc(C(C)C)[nH]3)C2)=O)cc1 N1(C(Cc2nn(C)c(Cl)c2)=O)CCN(C(C2(C)COCCO2)=O)CC1C1CC1 N1(C(C=CC(C)(C)SC)=O)C(C(N2CCSCC2CO)=O)CCC1C1CC1 N1(C(C(CC)CC)=O)CC(C)CN(C(C2NC(=O)CC2C)=O)CC1C c1(CNC(C2CC2C(=O)Nc2ccn(C3CCC3)n2)=O)cccc(OCF)c1 c1(C(=O)NC(CCOC)CNC(=O)C(C)(C)C(C)C)cc(C)c(C)c2ncsc12 N1(C(COCCCC)=O)C2CCC1C(C(=O)NCc1nccc(O)n1)C2 CC(C)(F)C(C)(F)C(=O)NCC1CN(C(=O)CNC=O)CC1(F)F N1(C(C=CCNC(c2c(CC)nco2)=O)=O)CCC(OC)C(F)C1 C(c1cnn(C)c1)=CC(N1CC(C(N)=O)(CNC(C2CC23CCOC3)=O)C1)=O N1(C(C2(CC=C)CN(C(=O)C=Cc3ccncc3)C2)=O)CCOC2CC12 N1(C(c2n(C)ncc2I)C(=O)NCc2ccccc2)CCC2CCCCCC2C1 c1(Cn2c(NC(C(=O)NCC(c3ccccc3F)C)=O)ccn2)ccc(Br)cc1 C(=O)(C(C)CC(C)(C)C)N(CCC(C(C)C)NC(C1CCC(C)O1)=O)C C(CCCCC(=O)NC1C=CCCC1CO)N(C)C(C1CCOC1C1CC1)=O C(=O)(C(CNC(C1C2CC(=O)CC12)=O)CC(C)C)NCCc1cnc(C)s1 C(=O)(CS(=O)(=O)c1ncc[nH]1)N1C(C)C(O)CCC1.c12cccc(c1)OC2 C1(C)(C(=O)NCC2(NC(C(C)N(C(C)=O)C)=O)CCCCC2)CCCCCC1 C(=O)(C1=CCSC1)NC(CC)(C)CNC(c1cc(-c2ccc(Cl)s2)on1)=O Cc1cnc(F)cc1C(c1nnnn1CC1CC1)NC(CCO)c1cccs1 c1(CC(C(N2CC(F)(C(=O)OCC)C2)=O)F)ccc(OC)cc1 N1(C(CNC(C(CC)C)=O)=O)CC2CC1C2NC(C1CC1Cl)=O n1(C2(C(=O)N(CCC3CCC(N(C(CC)=O)CC)C3)C)CC2)cnc2ccccc12 Cc1cccc([N+](=O)[O-])c1N1CCC(C)C(NC(C2CC2C2CCCC2)=O)C1 Cc1cc(C(N2CC(=C(F)CNC(=O)CNS(C)(=O)=O)C2)=O)nn1C(C)C1CC1 CN1CCN(C(C2C3CCCCC23)=O)C(CNC(c2cnn(C)c2C(F)F)=O)C1 c1(C(=O)OCC(=O)CC2CC3CCC2C3)c[nH]c2cnccc12 c1(C(N2CC3C(C2)C3(F)F)=O)nc2ccc(-c3ccc(O)c(C4CC4)c3)cc2o1 c1(CC)ccc(CNC(=O)NCC2(O)CCCC2(C)C)c(OC)c1 c1(C(=O)NCCC(C)NC(c2ccc(=O)oc2)=O)occ2c1CCOC2 N1(C(C(C(C)C)SCC)=O)CCC(C)(C)C1C(=O)NCCCOC(C)=O C1(C(N2CCN(CC=C)CC2)=O)CCN(C(c2occc2C)=O)C(C)C1 C#Cc1cnc(C(=O)NCC(O)CN(C)C(C2CCCCO2)=O)c(C)c1 N1(C(c2ccc(OC)cc2I)=O)CC2CN(Cc3sc(C=O)c(Br)c3Br)CC2C1 C1(N(C)C(C2CCCN(C(=O)C(=O)NCC(F)(F)F)C2)=O)CCOC(C)(C)C1 Cc1nccc(C(=O)N(CC(C)NC(C2(C)CC2c2ccccc2)=O)C)n1 c1(C(=O)NC2(CF)CN(C(CCSC)=O)C2)cc(C(N)=O)cn1C C(C(C)C(F)C(=O)NCC1CCOCC1)NC(CN(C1CC1)CC)=O C(=O)(C1=NOC(C)C1C)N1CC(C(=O)NC(CC#C)CO)C(CCC)C1 N1(CCNC(c2coc(C(F)F)c2)=O)CCCN(C(C2CC2C2CC2)=O)CC1 C(C1SCCc2ccccc21)OC(CN(c1cc(C)c(OC(F)F)nc1)C)=O N1(C(C)=O)CCC(C(=O)N(C)CCNC(c2sccc2CO)=O)CC1 N1(C(C2CCOCC2)C(=O)NCCCOC)Cc2cccc(F)c2C1 C1(C(N2C3C(NC(C4(NC(=O)C5CC5)CC4)=O)C(C3)C2)=O)CC2(C1)CC(F)(F)C2 c1(OC)ccc(C(=O)NCCCN(C(=O)C=CC(=O)N(C)C)C)cc1OC1CC1 N1(C2CC2)CSCC1C(=O)NCCN(C(C(=O)OCC)=O)CC.c1cn(C)cn1 C1(C)(CNC(CCC(=C)C)=O)CN(C(c2nncn2CC)=O)C(C)(C)C1 C1(NC(C2=C(C)S(=O)(=O)CC2)=O)CN(C(C2CCCCO2)=O)C2(CCOCC2)C1 N1(C(c2c(CC)nccn2)=O)CCN(C(C2(O)CCC(CC)C2)=O)CC1C c1(C(N(CCCNC(=O)C=Cc2ccc(C(F)F)o2)CCO)=O)ccc(O)c(Cl)c1 C1(NC(C(C)OCC2CC2)=O)CCCN(C(c2cnc(Br)s2)=O)C1 c1(C(=O)NCC(C)(CO)NC(C2CCc3cnnn3C2)=O)cnc2sccc2c1 N1(CC(=O)OCc2cccc(C(C)C)n2)CCC2(CC1)CC2C(N1CCCC1)=O c1(C(N2CCC(NC(c3ccn(CCOC)n3)=O)(CF)C2)=O)cc([N+](=O)[O-])sn1 N1(C(CC2CC(OC)C2(C)C)=O)CC2CCC1CN2C(=O)CC1CCCCCC1 C1(O)(CNC(c2c(CC)cncc2)=O)CCN(C(=O)CSCC(N)=O)CC1 N1(C(C(C)=C2CCC2)=O)CCC2(CCN(C(c3ncccc3N)=O)CC2)C1 C(C(=O)N1CC=CCO1)NC(=O)CCc1cnccn1 C1(c2nc(CC(=O)OC(C)C(F)(F)F)[nH]n2)COC(C)(C)C1 N1(C(c2cc(C)n(C)n2)=O)CCC2(CC1)CC2CNC(C1CC(F)C1)=O N1(C(COCCC=C)=O)CCCCCC(NC(=O)C(C)Cc2ccccc2Cl)C1 C1(C)(CC(=O)Nc2c(C(=O)OC)con2)CCCN(CCN(C)C)C1 Cc1c(C(N2C(C(N3CC(O)C(F)C3)=O)CC3CC23)=O)cccc1I C1(NC(c2cc(CF)on2)=O)CC2CCC1C1CN(C(=O)C=C(Cl)Cl)CC21 CCCC(CNC(=O)CC1CCCC1O)C(=O)N1CCC(O)(C(N)=O)C1 CCC(C)CCC(=O)N1CCCC1C(=O)NC1(C)CCCC1(F)F N1(C(C(C=C)(C)C)=O)CCC2(CC1)CC2CNC(c1cc(C)nc(C2CC2)n1)=O S(=O)(=O)(c1ccc(NCC2CC2C2CCCC2)c(F)c1)NCCNS(NC)(=O)=O Cc1nn(CCO)c(C)c1NC(N1CC2CC1CN2C(=O)CC1CCOCC1)=O C1(C(=O)NC(C)CCC2CCCCO2)CC(O)CN1C(=O)OC(C)(C)C N1(C(=O)NC)CC2CC1C2C(N1CC(NC(c2cn(CCO)nn2)=O)C(O)C1)=O C1(C(C(C)C)NC(c2ccn(C)n2)=O)CCN(C(C2C(C#N)C2(C)C)=O)CC1 c1(-c2cnc(CNC(C3CCSCC3)=O)nc2)ccc2c(c1)CCC2=O Cc1nnn(C)c1C(=O)NCC1(O)CN(C(C2CCC=CCC2)=O)C1 CC(C)C(C(C)NC(=O)Cc1cnsc1)NC(=O)CCc1cncc(F)c1 CC(C)(C(=O)NC1CC1NC(c1cc(CCO)on1)=O)c1cccnc1 N1(C(c2cnc(OCC)nc2)=O)CC2(CC2)CC1C(=O)N(C)CC#N Cn1nc(C(=O)NCC2COCC2NC(C2(C)COCCO2)=O)cc1C(F)(F)F N1(C(C2ON=C(CC)C2)=O)CCC2(CC(NC(=O)CCOC3CCCC3)C2)C1 CCC(C)(COC)C(=O)NCC(C(=O)N1CC(C)(CO)C1)N(C)C Cc1nn(CC(=O)NC(C)(CNC(=O)C(C)C2CCCC2)C(C)C)c(=O)o1 C1(C)(C(=O)NCc2cc(C(=O)NCC3C(OC)CCC3)n(C)n2)CCC(=O)NC1 C(=O)(CC(C)CC(C)C)NCC(C1N(C(COC(C)=O)=O)CCC1)(C)C c1(C(N2CCCC(CNC(C3CN4CCN3CC4)=O)C2)=O)cnc2[nH]cncc1-2 C1(CCC)CCCN(C(=O)CCCCNC(=O)C(O)CC(C)C)CC1 N1(C(C2C(O)CCN(C(c3nccnc3Br)=O)C2)=O)CCOc2ccccc2C1 CC(CN(C)C)CCC(=O)N1C2CCC1C(CNC(c1cc([N+](=O)[O-])n[nH]1)=O)C2 c1(C(N2CCN(C(C(N)=O)=O)CC2C2CCC2)=O)nc2c(Br)cccn2n1 Cc1c(Cl)nc(CC(C)C)[nH]c1=NCC(C)(C(C)C)NC(=O)C(F)C(F)(F)F O=C(C1=C(Cl)CCCC1)NC1CCC(O)CN(C(C2CCC(CO)CC2)=O)C1 CC1CN(C(=O)CC(F)F)CC1NC(c1cncc(-c2ccccc2)c1)=O C(N=c1[nH]c(=NCCCC(=O)N(C)C)c2sccc2[nH]1)C1(OC)CCOC1 CC1CCN(C(c2csc(Cl)n2)=O)C1C(=O)NCC1(CO)CC(C)C1 c1(C(N2CC3C(CNC(C(C4CCC4)OC)=O)C3C2)=O)cncc2ncn(C)c12 N1(C(=O)CC23CCC(CC2)C3)CC2(C=C(C(=O)N3CC4C=CC3CC4)CO2)C1 C1(N(C(C(CCOC)NC(=O)C(C)=CC(C)(C)C)=O)C)CC2CCC1CC2 c1(C(N2CCC(O)(CCNC(CCSCCC)=O)C2)=O)cc2n(n1)CCOC2 N1(OC)CCCC(C)S(=O)(=O)CC1.c12nccc(n1)-c1cccc(c1)-c1nccn1-2 c1(SC)cc(CNC(C2(CN(C)C)CC2)=O)cs1.C12(CC1)CC(=O)NC2 Cc1cn2cc(CC(=O)N(CCNC(C3(CO)CCCO3)=O)CC3CC3)nc2s1 c1(CC(=O)NCC(C)NC(CCCCSC)=O)ccc(F)cc1[N+](=O)[O-] CC(O)CCCCCC(=O)NC1CC2(C1)CC2NC(c1ccn(C(F)F)n1)=O C(=O)(C1CCOc2ccc(Cl)cc21)NC1C(CNC(C2CC(C#N)C2)=O)CCC1 C1(C)(CNC(CCSCC)=O)CN(C(c2ccc(C(=O)OC)o2)=O)C(C)(C)C1 CC(=Cn1ccnn1)C(=O)NC1(CNC(C2(C#N)CC2C(F)(F)F)=O)CC1 C1(CNC(c2cnccn2)=O)CCN(C(c2ccc3cc[nH]c3c2)=O)CC1(F)F n1(CC)nnnc1C(C1CCCO1)(C)NCC(C)COC(C)C c1(C(C)NC(=O)C(c2cccs2)NC(c2cc[nH]c2)=O)cccc(O)c1 N1(C(C2=CC(C)(C)C2)=O)CCCC2(CCN(C(C34CCCC(C)(C3)OC4)=O)C2)C1 C1(C(=O)NCC2=C(C)CCC2)C2CC(O)C(C2)N1C(c1ccc(C)cc1F)=O N1(C(C(CCSC)NC(N)=O)=O)CCN(C(c2nccn2C(C)C)=O)CC1C C(=O)(CC1OCCc2sccc21)N(C)Cc1cn(Cc2ccnc(Br)c2)nn1 C1(C(C(=O)N(CCCC)CCOC)C)CCn2cncc2C1 c1(C(=O)NCC(C)(CC2CCC2)OC)c(C)cccc1F C1(C(N(CC(CO)(CO)NC(=O)Cc2ccc(F)cn2)C)=O)CC(=O)NC(=O)C1 S(=O)(=O)(c1cccnc1Cl)N1CC2(CC(NC(=O)Cn3cc(Br)cn3)C2)C1 N1(C(c2n(CC)ncc2)=O)CC(NC(=O)CNC(=O)CNC(C)=O)C2(CCC2)C1 C(=O)(CCCC(C)(C)C#N)NC(C(N1CC(O)(CN(C)C)C1)=O)CN(C)C N1(C(c2nc(CC)sc2N)=O)CCCC(F)(CNC(C2CC(CC)=NO2)=O)CC1 C1(C(=O)OC)CC(C(=O)NC(C)(C)CCNC(c2ncn(C)n2)=O)C12CCCC2 N1(Cc2cn(C(CC(C)(C)CO)Cc3cccc(Cl)c3)nn2)CC(=O)CCC1=O C12(C(=O)NCCCCNC(C3(C)CCC(C)C3)=O)CCC(C1)OC2C c1(NC)ccc(C(=O)N(Cc2cn(CC3CC3)nn2)CC2CCCO2)cc1F N1(Cc2c(OCC)cccn2)CCc2cc(CN)ccc21 N1(C(COCP(C)(C)=O)=O)CCN(C(c2nccnc2N)=O)C2CCC12 C1(C(=O)NCCCc2n[nH]c(C)n2)(CC)CCCN1C(=O)C(C)OC(C)(C)C c1(C(N2C(=O)CC(C(=O)NCCC(C(C)C)OC(C)C)C2)C)ccc(O)c(O)c1 C1(OCCNC(C(C)n2ccnc2)=O)CCN(C(C2C(C(C)=O)C2(C)C)=O)C1 CC(C)C(CC(=O)N=c1ccn(CCCO)[nH]1)NC(C1CCSC1)=O CCC(C)(CNC(C12CCCC1C2)=O)C(=O)NCC1(CO)CCCO1 C1(CCNC(C2(Cl)CC2)=O)CCCN(C(=O)CC2=CCCC2)CC1 CC1(C(N2CC(OCC(=O)NC3CCNC(=O)CC3)C2)=O)CCC(=O)NC1 C1(C2CC2)(COC)CN(C(=O)CN(C(=O)CC2CCC(C)O2)CC2CC2)C1 N1(C(C(C)(C)CCC#N)=O)C2CCCC1CN(C(=O)CC1CCCCC1(F)F)C2 C(=O)(C(C(C)C)NC(c1cccnc1CNC(C1C=CCCC1)=O)=O)OC C1(=O)C(F)C(C)CN1.C(=O)(C(C)(C)NC(=O)C=CCCC(C)C)OCC c1(COC)ccc(C(=O)NCC2(F)CC(NC(C3CC3C)=O)C2)s1 N1(C(c2ccc(CC)cn2)=O)C(C(=O)N(C2CC(O)C2)C)CCC12CC2 N1(C(C2(COC)C=CCC2)=O)CCC(C(C)(C)C)(CNC(=O)C=C(C)C(F)F)C1 N1(C(c2ccc[nH]2)=O)CCC2C(C1)CN2C(c1ccc(F)c(C(F)F)n1)=O C(=O)(C(C#N)C(C)(C)C)NC(CC)CN(C(c1cncc(COC)c1)=O)CC C(=O)(C(F)(CNC(=O)C(C)=C1CCCC1)C(C)C)N(CCCN(C)C)CC c1(NC)ccc(C)cc1C(N1CC(C(C)(C)O)(CNC(=O)C(C)(C)CO)C1)=O C1(CC)C(C(=O)NCCCCN2CCCC2)CCN1C(=O)CC1CCCC2CC12 C1(OC)CCC(C(=O)NCCCCCN(C)C(c2c[nH]nc2C2CC2)=O)C1 CCCS(=O)(=O)C(C)C(=O)N1CC2CN(C(C3(C)CC(C#N)C3)=O)CC2(C)C1 CCC(C(=O)N1CCC(CNC(C2CN(C(C)C)C2)=O)C1)OC C1(C(N2CC(C)(NC(c3ccoc3Cl)=O)C2)=O)CCC2CC1CO2 N1(C(c2cccc(C#C)c2)=O)CCC2CCN(C(=O)C=C(C)C#N)CC2C1 n1(CC=C)cc(C(=O)N(C)CC2CCCN2C(=O)C(C)N(C)C)c2ccccc12 C(=O)(C(C)(C)C(O)C(C)C)NC(CCCNC(c1c(CC)nco1)=O)(C)C C(c1cccc(Cl)c1)=C(C)C(=O)N(CC(C)NC(=O)CCC(C)O)C C(=O)(C1=C(Cl)CCC1)N(CC(C)NC(=O)Cc1cc(C)ccc1OC)CC Cc1ccc2cc(CN3CCC(O)CC3C(N3CCC(CO)C(O)C3)=O)sc2c1 N1(C(C=COCC)=O)CCC(O)(CN(C(=O)C(O)C(C)C)Cc2ccccc2)CC1 Cc1ccc(CS(N2CC(C)(F)C2)(=O)=O)c(F)c1 O=C(CCN=C(NCc1ccsc1)NCC1CCOCC1)NC1CCCCC1 c1(C(=O)NCC2(C(F)F)CCN(C(c3n(C)ccc3)=O)C2)cccc([N+](=O)[O-])c1 C(CC(=O)N(CCCCNC(=O)Cn1ccnn1)C)N(C(C)=O)C CC1CN(C(=O)CSCc2ccc(F)cc2)CCN1C(c1ccc(O)nn1)=O C(=O)(C1CNc2ccccc21)NCC(C)N(C(CC(CC)C)=O)C c1(C(C(=O)NC(CNC(CCNC(COC)=O)=O)C2CC2)O)cc(Cl)ccc1F C(=O)(CC1COCc2ccccc21)N(CC(C)(C)NC(C1CCN(C)C1)=O)C C=CCC(C(=O)N1CC(NC(C2CCCCCC2)=O)C(SC)C1)C(C)(C)C CC1CC(NC(=O)CCNC(C2CC(F)(F)C2)=O)CCN1C(c1ccccc1)=O CC(C)CC(O)C(=O)NCc1ncoc1C1CN(C(=O)CC(C)CF)C1 c1(C(=O)NC(CC(C)NC(c2nonc2N)=O)C)cc(S(=O)(=O)N(C)C)cn1C c1(CNC(=O)NCC(CN(CC)CC2CC2)O)nc(C2CC2)cs1 C1(NC(c2ccoc2Br)=O)CCN(C(c2cnns2)=O)CC12CCC2 C(C(C)C(F)C(=O)NCCCc1ccnn1C)NC(Cn1c(C)nnn1)=O C1(C2(C(=O)NCC(CNC(=O)CCC3OCCO3)F)CC2)CCCCO1 C12(C(=O)NC3C(CNC(C4CCCSC4)=O)CCC3)CC(C(F)F)(CO1)C2 Cn1cc2cc(CC(N3CCN(c4ccc(Cl)cc4)CC3)=O)ccc2n1 Cc1cncc(C(=O)NCCn2cc(CNC(=O)CC3CCCOC3)nn2)c1C c1(C(=O)NCCCCN(C)C(C2CC2(C)C)=O)nn(C)cc1Br Cc1ccn(CC(N2CCCC(NC(=O)CNC(=O)CN(C)C)C2)=O)c(=O)c1 c1(OCC)ncccc1NC(C1CCC(COC)CC1)c1nnnn1C1(C)CC1 c1(C(=O)NC(C2CN(C(C3CCC(F)CC3)=O)C2)C)c(Br)nc2n1CCCC2 C1(NC(C(C)Sc2ccccc2)=O)CN(C(c2nnc(S)n2C)=O)CC1N=[N+]=[N-] c1(C(=O)NC23CC(CNC(C(C)C#N)=O)(C2)C3)cccc(Cl)c1OC(F)(F)F N1(C(CCn2ncc(C)c2)=O)CCC2(CCCCC2NC(C2CCC2)=O)C1 C(C(C)CC(=O)NCCn1cnnc1)NC(C=CC(C)(C)SC)=O CC1CN(C(=O)NC2CCNCC2)CCN1C(=O)C(C)C(F)F.CC(F)(F)F N1(C(C(CC=CC)NC(=O)C(F)CCCCC)=O)CCC2CN(C)CCC12 c1(C(=O)NC(C2CCN(C(CCC(C)(C)OC)=O)C2)C)ccc2nnn(O)c2c1 c1(-c2cc(CC(C)(C)C)on2)nc(C2CCOCC2)nn1CCc1ccccc1 c1(C(C)(C)C)ncc(C(=O)NCC(C2CCC2)NC(c2n[nH]cc2Cl)=O)cn1 C1(NC(N(C)C)=O)CCN(Cc2cn(CCOCC3CCOC3)nn2)C1 c1(C(N2CCC(CCNC(C3C(C#C)C3)=O)CC2)=O)c(F)cc(C)cc1Cl C1(C(N(C2(C)CC2)C)=O)CC(C)(C)CN1C(C1OCCC1(C)C)=O N1(C(C(CC#C)O)=O)CC2C3CCC(C(NC(c4cncc(CC)c4)=O)C3)C2C1 C1(CNC(C2CCCCCC2)=O)CCCCN(C(C2(C(O)C(F)(F)F)CC2)=O)C1 c1(C(N2CC(C(C)C)C2)=O)cncc(CNC(=O)C(c2cncnc2)C)c1 C1(C(=O)OC)CN(Cc2cccc(NCc3cccnc3)c2)CC1c1cccs1 C12(NC(c3cc(CC4CC4)c[nH]3)=O)CCCC1CN(C(C1CC3CCC3C1)=O)C2 C(=O)(C(C)CCCOC)NCCCN(C(C1(C=C)CC1)=O)C1CC1 N1(C(C2(OC)CC(C)C2)=O)CCCC(CC(N2CCCC(N(C)C)C2)=O)CC1 C1(C(N2CCC(C)(NC(C(CCCC)C)=O)CC2)=O)CCc2c(ncn2C)C1 C1(NCCCCCC=C)CON(C(=O)OC(C)(C)C)C1 C1(CN(C(=O)OC(C)(C)C)CCO)CC2OC(=O)OC2C1.C12COCC1NC2=O c1(CC(=O)N(CC(C)N(C)C(c2cccc(CC#N)c2)=O)C)ccc(F)c(Cl)c1 CC(N=c1nc(N(C)CC2CC2(F)F)c2c([nH]1)COC2)c1ccoc1 N1(C(C2C(C(C)O)C2)=O)CCC(C)(CNC(c2ccnn2C2CCCC2)=O)CC1 C1(OCCNC(C2CCN2C(=O)CCc2ccoc2)=O)CC1(F)F Cc1cc(F)c(F)cc1NC(=O)CN1CCN(C(c2cnc(Br)o2)=O)CC1 C1(C(=O)OCC)CCCC12CCN(C(c1ccc(OC)cc1)C(=O)NC(C)C)C2 c1(C(C)C)nc(=NC2CN(C(c3cc(F)ccc3Cl)=O)CC2C)s[nH]1 CN1CCN(C(=O)C(O)CC2CCCC2)CC1C(=O)Nc1ccc(Cl)nc1 N12CCC3(CC3C(=O)N(C(C)C)CCC1=O)C2.N1(CCNC(N)=O)CCCC1 C12(CNC(CNS(N)(=O)=O)=O)CCC(NC(C3CC3C(N)=O)=O)(CO1)C2 C1(C)(NC(C2C(=C)C2)=O)CCN(C(c2oc(CO)cc2C)=O)CC1 N1(C(COC)=O)Cc2cnn(C3CCN(C(C4C(C(F)F)C4(C)C)=O)CC3)c2C1 c1(CN2CCN(S(=O)(=O)CC3CCC3)C3C2C3)c(F)cc(I)cc1F Cc1cnc2n1CCC(NC(C1(n3cccn3)CN(C(=O)C(N)=O)C1)=O)C2 CCCC(C(=O)N1CCCC1C(C)NC(=O)CC1CC2CC2C1)OC C1CC2(C1)CSCC2NCC1CNC2(CCC2)C1 CC1=NOC(C(=O)NC2CCN(C(c3[nH]nnc3C)=O)C2)C1 C1(CNC(C2=NNC(=O)C2)=O)CCC2CN(C(=O)CC3CS(=O)(=O)C3)CCC2C1 C(CC(=O)N1Cc2ccccc2CO1)NC(C1(C)CCCO1)=O c1(C(C)C)ccc(C=CC(=O)NC2CCC2NC(C2CCCN2C=O)=O)cc1 Cn1ncc(CNC(C2CC2(F)F)=O)c1C(=O)NCCOCC(F)(F)F Cc1cc(C(=O)NCC(C)(C(C)C)NC(=O)Cc2ccc(Cl)cc2Cl)nnc1C C1(C(F)F)(CNC(C(C)OCC#C)=O)CCN(C(c2cn(C3CC3)cn2)=O)C1 c1(N2C(=O)CC(NC(C(=O)OCC)CCN(C)C)C2)ccc(OC)c(Cl)c1 c1(C(=O)NC2CC(NC(C3CN(CC)C(=O)N3)=O)C2)cc(C)c(O)c([N+](=O)[O-])c1 c1(C(=O)NC(C)CCNC(=O)CSc2nc[nH]n2)c(O)cc(Cl)cc1F Cn1c(C(N2CCCC2CC(=O)NCCc2nn[nH]n2)=O)cc2ccccc12 c1(N2CCCC(C)(OC)C2)[nH]c(=NCc2ccc(C)cc2Br)nc2sccc12 CCC(C)C(C(=O)NC12CCC(NC(=O)C(C)OC3CCCC3)(CC1)C2)N(C)C c1(C(=O)NC2CCN(C(C3CCCC4CC34)=O)CC2F)cc2ncccc2[nH]1 C1(C(C)CNC(c2ncccn2)=O)CCN(C(C2(N(C)C)CCCC2)=O)CC1 C#CC12CCC(C(N3CC4CCC3C4NC(=O)CCCCCC=C)=O)(CC1)CC2 C1(CC(=O)NCCN(C(C)C)C)CCCC1NC(=O)CSCCC#N C(=O)(C(C)(C)CCSC)N1CCN(C(c2cn(C(C(=O)OCC)C)nn2)C)CC1 C1(NC(CC(CC)C)=O)CN(C(=O)NC2(Nc3cccc(C)c3)CC2)CC1(C)C c1(C(=O)NCC(CO)NC(C2(C)CC3CCC(C2)S3)=O)c[nH]c2c(Cl)cccc12 c1(OC)ccc(NC(C2CCN(C(=O)C(C3CCOCC3)F)C2(C)C)=O)c(O)c1 CC1CCCC=C1C(=O)N(C)CC1(O)CN(C(=O)COc2ccccc2)C1 N1(C(c2c(C)cccc2)=O)CC(C2CCCCN(C(C3CCCS3)=O)C2)C1 N1(C(c2ccoc2)=O)CCn2cnc(-c3csc(CO)c3)c2C1 C1(C)(C)CC(=O)N1.c1(C(C(N2CC(CCCCNC(C)=O)C2)=O)C)cccc(F)c1 C(=O)(C(CNC(=O)CCc1cncnc1)CC1CC1)NC(c1ncc[nH]1)C S(=O)(=O)(c1cnccc1N1CCCC(C#N)C1)N1CCCC(CC(=O)NC)C1 Cc1ccc(C(=O)NC2CN(C)C2)c(-n2cc(C(c3ccc(Cl)cc3)O)nn2)c1 C1(N(C(c2ccc(C(=O)OC)s2)=O)CC)CCCN(C(=O)Cc2sccc2Cl)C1 c1(CNc2cccc(C(=O)NC(C)C(=O)NO)c2)ccc(O)c2ccccc12 CC1(C)CN(C(c2csc(CO)n2)=O)CC2(CN(C(C3C4CC5C(C4)C35)=O)C2)O1 C1(C)(C(N2C(C(=O)NCC(C)NC(=O)OC)CCC2)=O)CNC(=O)C1 Cc1cc(C(=O)N(C2CCN(c3ncncc3Cl)C2)C)n(-c2ccccn2)n1 c1(OC)ccnc(C(=O)N(CCCN(C)C(c2coc(SC)c2)=O)C)c1N c1(C(N2C(CNC(C3CC(SC)C3)=O)COCC2)=O)ncc(C)cc1C N1(C(C(C2CCCC2)OC)=O)CCN(C(=O)C(C)OC(C)=O)CC1 C(=O)(C1=CCCC1(C)C)N1CCC(NC(c2cnc(OC)nc2)=O)C12CC2 CC(C)(C#N)CCC(=O)N1CCC(CCNC(C2(C)CC2c2ccccc2)=O)C1 c1(NC(c2ncncc2Cl)=O)ccc(N2CC(OCCO)CC2)nn1 N1(C(CC2C(CC)C2)=O)CCOC(C(=O)NCCC2=CCOCC2)CC1 CC1(C)CCN(C(=O)C(O)c2cnc[nH]2)CC1NC(=O)CCOCC(F)F CCC(C)(CNC(=O)C(C1(O)CN(C(C2CCC(F)CC2)=O)C1)F)C(N)=O C1(C)(CNC(c2c(C)csc2)=O)CCCN(C(c2cc(C)sc2C)=O)C1 N1(C2(C(N(CCN(C(C3CC(OC)C3)=O)C)C)=O)CC2)CCOCC1 c1(C(N2CCC(N(C(=O)C3=COCCO3)C)C2)=O)ccc2cccc(Cl)c2n1 C1(C)(C(N(C)CC2(N(C)C)CC2)=O)CCN(C(=O)CC2CCCC3CC23)C1 c1(C(=O)NCC(C)NC(c2cncc(C)n2)=O)sccc1S(=O)(=O)N1CCCC1 c1(C(=O)NC2(CCNC(CC3CCN(C)C3=O)=O)CCC2)nccc2occc12 C(CC(C(=O)NCC=CCNC(=O)Cn1nnc(=N)[nH]1)OC)OC n1(CCOC)nc(C(=O)NCC(C)(CO)NC(C2CCC(C)(C)O2)=O)ccc1=O C1(C(=O)NCC(CN(C)C(c2csc(C(F)F)n2)=O)O)Cc2cc(Cl)ccc2O1 N1(C(c2ccc(SCC)cc2)=O)CCN(C(=O)CCc2ccncn2)C(CF)C1 C#Cc1cccc(C(N2CCCC(C(=O)NCC(C)C(F)F)CC2)=O)c1 c1(OC)cc(C(=O)NC(CNC(c2nc(C)oc2C)=O)CO)ccc1[N+](=O)[O-] C1(NC(C2(C)CC(=C)C2)=O)CC(C(=O)N2CCSC(C)C2C)=CC1O C1(CNC(C(F)=C(C)C)=O)CCCN(C(C2CCCCS2)=O)C1 N1(C(Cc2ccc(C)s2)=O)CC(CNC(C2CCCS2)=O)CC(C)C1 C(=O)(CCCCCNC(=O)CN1CCCC1)NC(CCC(=C)C)C c1(NCC(CNC(c2cc(SC)ncc2)=O)C)nc(C(F)(F)F)ccc1C#N c1(C(N2C(C)C(NC(C3CCC=CCC3)=O)CC2)=O)c2c(c[nH]c1=N)CCC2 c1(C(=O)NC(CNC(=O)CNC(N2CCCC2)=O)C2CCC2)cnnc(O)c1 C1(C2C(CC(=O)N(CCNC(C3CC(CC)C3)=O)C)C2)CCCCO1 c1(N2CCN(Cc3ccc(C#N)nc3)C3C2C3)ncc2ccc(F)cc2n1 N1(C(CSCCN(OCC)CC)=O)CCC2CN(CC(=O)NC3CCCC3)CC12 N1(C(c2c(N)cccc2Cl)=O)CCC2C(CCCN2C(=O)C=CC2CCCC2)C1 C(=O)(C1=CCCOC1)N1CC(F)(CNC(=O)CCCn2cncn2)C1 c1(CC(=O)N(CC(C)NC(C(C)OCCOCC)=O)C)sccc1C C12(C(N3CCC(NC(c4cc(F)cs4)=O)C(O)C3)=O)CCCCCC1OCC2 C1(CC(N2CCC(CCNC(CCOC(C)=O)=O)C2)=O)C=NN(C)C1=O.C c1(C(C)C)cc(C(N2CC(CCNC(=O)CC(C)(F)F)C(C)C2)=O)ccc1F N(C(=NCCC=C)NC1CCC12CCC2)C1(CC#C)CCC1 c1(CC(=O)NC(C)CCNC(C2CCCC2(F)F)=O)ccc2c(c1)CCCN2C N1(C(c2c(C)sc(Br)c2)=O)CC2(CCN(C(C3(C(=O)N(C)C)CC3)=O)C2)C1 Cc1nc(C)n(CC(=O)NC(C(=O)NC(c2ccco2)CO)C2CCCO2)n1 C(=O)(CCCCCC1CC1)NCC(C)NC(c1cn(CC2CCCO2)nn1)=O N1(CC(=O)N(CCC)C(C2CC(C)C2)=O)C2CCC1CN(Cc1cccs1)CC2 Cc1cc(N(C)CC2CCOCC2)nc(=NCC(C)c2ccc(Cl)cc2)[nH]1 c1(C(N2CCCC(C(C)C(=O)N(C(C)CN(C)C)C)C2)=O)cncc2[nH]ccc12 C1(C)(C(N2CCC(CC=C)(NC(=O)Cc3n[nH]c(=N)s3)C2)=O)CCCCNC1=O N1(C(C(C2CCN(C(c3nc(C)oc3)=O)C2)F)=O)CC2(CNC(=O)C2)C1 C1(C(N(C)CCN2CCCC2=O)=O)CCN(C(=O)Cc2cccnc2O)CC1 C1(c2n(CCC)nnn2)(OC(CNC(c2ccccc2)=O)=O)CSC(C)(C)C1 c1(C(=O)OC)n[nH]c2ccc(-c3nn[nH]n3)cc12.c12sc(cc1C)C(C)NC2=O c1(C(=O)NC(C(C)C)CNC(=O)CC2CCCCO2)cc(F)cc(Br)c1O C(CC(C)C(=O)NCC(O)CNC(c1onc(C)c1C)=O)=CCC N1(C(C2(C)CCC2)=O)CCCC(C2CCN(C(=O)CC3CCCOCC3)C2)C1 CN(C1CCc2cc(F)ccc21)C(=O)CC1CC(=O)C1 N1(C(c2ccc(C(C)C)s2)=O)CCC2CN(C(c3cccn3C)=O)CCC2C1 Cc1ccc2c(c1)C(C(=O)NCCN(C(C1CN3CCCN1CC3)=O)C1CC1)CC2 C=CC(C)(C)C(=O)NC1CC(NC(c2cnn(C(C)CC)c2C2CC2)=O)C1 C1(NC(=O)CC2CC(F)CN2C(C2CCCC2)=O)CC2(CCCCO2)C1 Cn1cc(C(=O)NCCN2CCN(C(C3CCC(C)(C)C3)=O)CC2)cc1Br CCCS(=O)(=O)CC(=O)N1CCC(NC(=O)CC2CC3(CC3)C2)C(CO)CC1 N1(C(C2(CC#C)CC2)=O)CCN(C(=O)C(C2(O)CCCC2)F)CC(O)C1 c1(CC(=O)NC2CC(CNC(c3c(C)ccc(O)c3)=O)C2)ccc2c(c1)COC2 c1(COC(c2ccc(CNC)cc2)=O)cccc2cncn12.CC1(C)CC1(Cl)C(=O)N C12(Nc3nc(C)nc(C(F)(F)F)c3)CCCC1CN(C(c1cn(C)cn1)=O)C2 c1(CC(C(=O)NCC(CC)(C)NC(c2cc(C3CC3)[nH]n2)=O)O)ccc(Cl)cc1 C1(C(=O)NC2(CC=C)CCN(C(=O)Cc3cnns3)C2)CCn2ccnc2C1 C12(NC(C(N3C(CC)CCC3)=O)=O)CCC1CN(C(=O)Cc1ccc(F)cn1)C2 N1(C(C(C(CC)O)C)=O)CCC2(CC1)CN(C(=O)CS(=O)(=O)CCO)CC2CO c1(OC)ncc(F)c(NC2CC(C(C)(C)C)CN(C(=O)OC)C2)n1 C1(CC)(NC(=O)CCCn2ccccc2=O)CCCN(C(=O)CC2CCOC2)C1 c1(CC(C(=O)N(CC(C)NC(COCCC=C)=O)C)O)c(F)cccc1Cl O=C(CCCCCO)N1CC2(CC2C(=O)NCC(F)CO)C1 C1(C(N(C(C)CCNC(=O)CSC(=N)N)C)=O)Cc2ccccc2CO1 C1(CC(=O)NC2(CNC(c3cc(OC)c(O)nc3)=O)CC2)CCCC2(CCC2)O1 Cc1cc(=O)n(CCC(=O)NC2CCN(C(=O)C3=CCCCO3)C(C)C2)cn1 c1(CCNC(c2ccncc2Cl)=O)ccc(CNC(C23CCC(C2)C3)=O)cc1 c1(C2(C(=O)NCCC3(O)CN(C(=O)C=C4CCC4)C3)CC2)ccc(F)cc1F CCC(C)C(C(=O)NCCc1cn(C)nn1)NC(=O)C(CSC)OC c1(C(=O)NCC(CNC(C2C(C)C2C)=O)F)cccc(-c2cccc(Cl)c2)c1 c1(CCNc2c(C)nn(C3CC3)c2)cc(F)cc(Br)c1 c1(C(N2C(CNC(C3CC(F)(CO)C3)=O)CC(OC)C2)=O)cc2cccnc2o1 c1(C(N(CCCOCCOC)C)=O)cc2nc(C)cc(C(F)(F)F)n2n1 c1(C(=O)NCCC2(C)CCN(C(C)=O)C2)ccccc1S(=O)C(F)(F)F C1(N(c2cc[nH]n2)C(c2cccnn2)=O)CCC12CCNCC2 c1(OC)ccc(C)c(C(=O)NCC(C)(C)CNC(=O)Cn2cc(C)ccc2=O)n1 c1(C(=O)NC2C(CC)CN(C(C3(CC(C)C)CC3)=O)CC2)c(N)cc(F)cc1F C=CCCCC(C(=O)NCCC(F)(F)Cl)NC(C1CCCCC1(C)C)=O CC1C(NC(=O)CS(=O)(=O)N(C)C)CCCN1C(c1nc(Cl)ccc1N)=O N1(C(=O)CCN2CCC2)CCC2(C1)CN(C(C1(c3cc[nH]n3)CC1)=O)C2 S(=O)(=O)(c1ccc(N2Cc3ccncc3C2)cc1Cl)NC(c1cn(C)cn1)C c1(OCC(=O)N(C)CC2(O)CN(C(C(C)OCC3CC3)=O)C2)cccc(F)c1 C(=O)(CCCC(C)(C)NC(=O)C(C1CCCC1)SC)NC(CC#CC)C C(=O)(CC(C)C(=O)NCCOC1CCN(c2ccnc(C(C)(C)C)n2)C1)OC c1(C(=O)NCCCN(C(COCC(=O)NC)=O)CCO)cnn2c1CN(C)CC2 c1(C(=O)NC2CCCC(NC(CC3C(C)CCC3)=O)C2)ccc(O)c(F)c1 C1(CC(N2CC(OC)C(OC)C2)=O)CCC(N=c2nc(SC)c3nc[nH]c3[nH]2)CC1 c1(CC)ccc(N(C(=O)CCCCC2CC2)CCNC(C2CCCC2CC)=O)c(C)c1 Cc1ccn(C(C)C(=O)N(C2CC(C(=O)NCC3(CC(C)C)CC3)C2)C)n1 c1(CC(=O)NCC(COC)C)cc(Cl)ccc1C C(=O)(C1=C(C)OCCC1)N(CC(C(=O)NCCCNC(=O)NC)(C)C)C C1(CNC(CCC=C)=O)(CO)CCCN(C(=O)C(C2CC2)OCC)C1 C(N=c1[nH]cnc2[nH]ccc12)C1N(C(C2CCCCC2OC2CCC2)=O)CCC1 C1(C(N(C)CC2(CC3CC3)CC2)=O)CCCC12CCN(C(C1(C)CCC1)=O)C2 C1(C(C(N2CC(C(=O)OC)(SC)C2)=O)C)CCCN(C(c2csnn2)=O)C1 N1(C(C=CCOC)=O)CCC(F)(F)C(CNc2nccc(CC(=O)OC)n2)C1 C(=O)(CCCS(C)(=O)=O)N1CC(CC(CNC(C2CN(C(C)=O)C2)=O)(C)C)C1 N1(C(c2cn(CCC)nn2)=O)CC2CC(C(=O)NCCC3CC(C)(C)C3)CC2C1 C(=O)(C1CCc2ccccc21)N1C(CN(C(c2ns[nH]c2=O)=O)CC)CCC1 C1(O)(CNC(COCC)=O)CCN(C(=O)Cc2coc(-c3cccs3)n2)C1 c1(C(N(CCC(C(C)C)NC(=O)C#CC(=O)N(C)C)C)=O)cccn2ncnc12 N1(C(C(C)(CO)NC(C(CCCC#C)C)=O)=O)CC2(CCC(O)CC2)C1 N1(C(CC=C)=O)CC2CC1CN(C(=O)C=CC1CCOCC1)C2 c1(N(C)C)ccc(C(=O)NCCC2(CNC(=O)C=CC3CC3)CC2)cc1 CC(C)(CO)C(=O)Nc1cccc(NC(=O)Cc2ccn(C(F)F)n2)c1 C(=O)(C(C#N)(CC)CC)NC(CCC)CNC(=O)CSc1nnnn1C c1(N2CC3C(C)C3C2)[nH]c(=NCCC2CCCCO2)nc2scnc12 C1(CNC(CN(C)S(N)(=O)=O)=O)CCCCCN1C(c1cc(=O)cc(Cl)[nH]1)=O c1(C(=O)NCCOCCn2cc(-c3c(C)ccs3)nn2)ccc(C(C)F)cc1 O=C(C1=CCCOC1)NC1CC(CNC(c2cnn(C3CC3)c2Cl)=O)C12CCC2 C1(C(=O)NCc2cnc(C)o2)CCN(C(=O)C2CCC3(CCC3)C2)O1 C1(CNC(C(=Cc2ccccn2)C)=O)C2CCC(C2)N1C(C1CN2CCC1C2)=O C1(C#CC(=O)NCC(C)CN(C(=O)C=Cc2ccc(Cl)cc2)C)(CC)CC1 N1(CCC(=O)NCCC2CN(C(=O)CC3CC3(Cl)Cl)C2)CCCCC1=O CC#CCC(C(=O)NCC(C)C(C)CC)NC(c1n[nH]c(C)c1Cl)=O N1(C(C=C2CCC(C)C2)=O)CCCC2(NC(=O)CSc3n[nH]c(O)n3)CCCC12 c12ccc(Br)cc1C(=O)O2.N1(CCSC2(OC(C)C)CCCC2)CCN(C)CC1 CC(C)C(C)C(C)CC(=O)N1CC2CC1C2NC(C1CCN(C)C1=O)=O C1(NC(C=Cc2nnc(C(C)C)o2)=O)CCN(C(=O)CSC2CC2)CC1O C#CC1CN(C(C2CCC(=O)N2)=O)CCN1C(=O)CCC1CC1(F)F c1(C(N2CC(C=C)C(NC(=O)C3CC3)C2)=O)nnc2ccccc2c1N C1(CNC(CC=C=C)=O)CN(C(=O)C(C)Cc2cnc[nH]2)CCCO1 c1(C(C(=O)NCC(n2cc(C3C4COCC34)nn2)C)O)cccc([N+](=O)[O-])c1 C1(C(NOCCCN(C)C)=O)CCCCC1NC(C1CC(=O)CCO1)=O C=CCCCC(C(=O)N1CC(O)(C(=O)NC(C(=O)C(N)=O)C)C1)NOC c1(OCCC#C)ccc(C(N2CCC(O)(C(C)NC(=O)CCC(=C)Cl)C2)=O)cc1 C1(CC)C(C(=O)NC(COC)C2CC2)CCN1C(c1nnsc1C)=O Cc1ccc2n[nH]cc2c1C(=O)NCC(O)CN(C(=O)C(F)(F)C(C)O)C c1(C(=O)NC2C(NC(c3csc(CO)n3)=O)COC2)c[nH]c2ccncc2c1=O C1(C(=O)N(C2(C=O)CC2)CC#N)OCCC1NCC(F)(F)F.CC(C)(C)O C=CCCC(C)C(C(=O)NCC1CCOC1)N1CC(C)OCC12CCC2 C(CN=C(NCc1cnccc1C(F)(F)F)NCC1CC1(F)F)OCC=C CC(=O)CCCC(=O)N1CCC(CN(C(=O)C(C)OCc2ccncc2)C)C1 C1(OC)CN(C(=O)Cn2ccc(C(F)(F)F)n2)CC1NC(C1CN(C(C)C)C1)=O c1(-c2cccc(CNC(c3n(C)cc(I)c3)=O)c2)ccn2c(O)nnc2c1 N1(C(Cn2ccc(C)cc2=O)=O)CCC2CCC(C1)N2CC1CCS(=O)(=O)CC1 c1(OC)ccc(CNC(c2[nH]ccc2CNC(=O)C2=CCCC2)=O)cc1F c1(CC)cccc(C(N2CC(CO)(NC(=O)C=Cc3ccc(Cl)cc3)C2)=O)c1N c1(C(=O)NC(C)CCCNC(C2(O)CC(C)(C)C2)=O)c[nH]c(=N)nc1O C1(C(C)C(=O)OC2(CO)CN(C(=O)OC(C)(C)C)C2)CCC(=O)NC1 C1(C(N2CC(CNC(c3cncc(C(F)F)c3)=O)C(C)C2)=O)(CC)CCOCC1 Cc1ccc(CN2CCC(N(C)C(c3ccc(-c4cc[nH]n4)s3)=O)C2)cc1 N1(C(c2n(CC=C)ccc2)=O)CCCCC1CCNC(C1CC1OC(C)=O)=O c1(C(=O)NC2C(OC)C(O)C2)c(CNC(C23CSCC2C3)=O)nnn1C C1(OCC(=O)NC(C=C)C2CC2)CCN(C(c2csc(O)n2)=O)C1 c1(C(N2C(CNC(CCC#CC)=O)C(C)CC2)=O)cc(OC)cc2ccoc12 c1(OC)cc(CC(=O)NC2CCCN(C(c3nccnc3N)=O)C2C)cc(F)c1 C1(NC(C(C)OCC)=O)CC2(CCN(C(=O)CS(=O)(=O)NC3CC3)C2)C1 C1(c2cn3nc2C3)CC2CCC1CC2.CON(C)C1CC1Cc1nnc(SC)o1 N1(C(CONC(=O)OC(C)(C)C)=O)CCCC12CCN(C(=O)CP(C)(C)=O)CC2 c1(CC(C(=O)O)NC(CNC(Cn2c(C)nnn2)=O)=O)ccc(O)c(O)c1 C#CCCCCC(=O)N1CCCC(C)C1CNC(c1cc(Cl)ncc1O)=O C(=O)(CC(=O)OCc1[nH]nnc1Cc1ccccc1)OC.C1C(C2CC2)NC1=O n1(CC(=O)N(CC(C)O)CCNC(=O)CCCc2ccsc2)cccnc1=O c1(C(N2CCC3(NC(C=CSC)=O)C(C2)C3)=O)sc2ccccc2c1Cl c1(CCC)ncc(C(=O)NC(c2ccccc2)CNC(c2cnnn2C)=O)s1 C12(C(N3CC(C)C(N(C)C)C3)=O)CC(CO1)N(C(=O)CC1(O)CCCC1)C2 C(=O)(C(CC(C)C)C(C)C)NC(N1CCN(C(=O)C(F)C(C)C)CC1)CCCCC C1(NC(C2CCC(CNC(COCC(=O)NC)=O)CC2)=O)CCC(C)NC1=O c1(C(=O)NC2C3CN(C(C(COC)(C)C)=O)C2C3)cc(C(F)(F)F)cc(Cl)c1 C1(C(=O)NCCN(OC)C)CN(C(C23CC(C#N)(C2)C3)=O)CC1C c1(N2CC(CNC(CC(CCC)CC)=O)C(F)(F)CC2)ncc([N+](=O)[O-])cc1F N1(CCCNC(CC2CC(=C)C2)=O)CCN(C(=O)C=C(CC)CC)CC1 C#CCC(CC#C)C(=O)N1CC2(CC2)CC1CNC(C1(C2CC2)CC1)=O N1(C(c2nc(CC)oc2)=O)CC(C)(C)OCC1CNC(c1csnn1)=O c1(OC)ccc(CN=c2nc(C3(C)CC3)o[nH]2)cc1C Cc1cc(F)cc(C(N2CCC2CNC(=O)CSc2nncs2)=O)c1C CC1(CC(N2CCOCC(NC(C3CCCCC(=O)N3)=O)C2)=O)CCCCCC1 C1(CNC(c2c(COC)ncs2)=O)C2CN(C(C3(C)CCCCC3)=O)CC12 C1(C(=O)NCC(CC)O)CN(C(=O)C(O)CN(C)C)CCO1 C=CCC(C)C(=O)NCCN(CCOCCO)C(c1coc(C2CCCC2)n1)=O CC1=C(CNC(c2ncsc2C)c2nnnn2CC2CCCO2)CCC1 N1(C(c2n(CC)ccn2)=O)CCC(C2(NC(=O)CCc3cncc(F)c3)CC2)C1 C(=O)(C(CCCCC1CC1)N(C)Cc1ccc(Cl)s1)NCCOC C(C(C)(C(=O)N1CCC(C)(CCO)C1)NC(c1cocc1C)=O)SC Cc1nn(C)c(C)c1C(=O)C(N1CCCC1CNC(c1csc(C(C)C)n1)=O)=O c1(C(=O)NCC(C)NC(C2(NC(C)=O)CCC2)=O)cc2ncn(C)c2cn1 Cc1cnc2c(C(=O)NCC3CCCC(NC(=O)CCCC#N)C3)cnn2c1 N1(CC(=O)N(CC(=O)N(C(COC)=O)C(C)(C)C)C)Cc2c(F)ccc(F)c2C1 CCCC(C#N)C(=O)NC(CC1CC1)C(=O)NCc1ccnc(F)c1 c1(C(=O)NCC(C)(C2CC2)NC(C(C)c2cccs2)=O)nccc2ccncc12 C1(C(N(C(C)CCNC(=O)CSc2ccccc2F)C)=O)CCOC2(CCC2)C1 c1(C(=O)NC2C(NC(Cc3cn(C)nc3)=O)CS(=O)(=O)C2)c(N)c(F)cc(F)c1F c1(-c2n(-c3ccc(F)c(Cl)c3)nc(C(F)F)n2)ccc2ncccc2c1 c1(C(=O)OC)ccc(C=CC(=O)NCCN(C(=O)CCCCN2CCC2)CC)o1 c1(C(=O)NC2(CNC(C(CC=C)C)=O)CCC2)cc(C)cc2c(C)ccnc12 c1(OC)ccc(Br)cc1C(=O)NC1CC(Oc2cc(N3CCCC3)nc(Cl)c2)C1 C1(C(=O)NC2C(CNC(COc3cn(C)nc3)=O)CC2)CC2C=CCC(C1)C2 c1(C(C(=O)NCC=C)N(CC)Cc2cn(C)nn2)ccc(-n2cc(Cl)cn2)cc1 C=CCC(F)(F)C(=O)NCC(C)C(F)C(=O)N1CC(CO)(CF)C1 C1(CNC(=O)Cc2cccs2)CN(C(=O)COCCO)CC12CC2.C1CCOC1 N1(C(C2C(CNC(C3N(CC)CCCC3)=O)CC2)=O)CCC2(CNC(=O)C2)C1 C(c1sccc1C)=CC(=O)N(C(C(=O)OC)Cc1c[nH]nc1O)C1CC1 N1(C(C2C(NC(c3c(C)scc3)=O)CCC2)=O)CC2COCC2C1 C(=O)(C(C(C)NC(C1CCN(OC)CC1)=O)C(C)C)N1CCC(O)(CC=C)CC1 C(=O)(C(C(C)C)N(C)C)NCCC(=C)CNC(C1CCN(S(=O)(=O)CC)CC1)=O C#CCCC(O)C(=O)N1CCC(C(C)NC(c2conc2C(C)C)=O)CC1 Cc1cccc(C(C)NC(C2(CNC(=O)CCn3cccn3)CC(C)(C)C2)=O)c1 C(C(C(=O)N1CCCCC1CN(C)C)C(C)C)NC(CCCOCC)=O Cc1c(C(=O)NCCC(C)NC(c2c[nH]nc2C(F)(F)F)=O)oc2ccccc12 C=CC(F)(F)C(=O)N(CCCNC(=O)C(O)Cc1ccccc1)C1CC1 c1(C(=O)NC2C(CNC(C(CSC)C)=O)C2)ccc(C)c(C#N)c1 c1(CC(=O)NCCNC(CCCCOC)=O)nc(Br)n2c1CCCC2 C(=O)(C(C)(C)CC(=O)N(C(C)CCNC(=O)CC(C)NC(N)=O)C)OCC C=C=CCCC(=O)N(C)CCN(C(=O)CC1CC(=O)NC1=O)C C1(CNC(C2N(C(C3(OCC)CCC3)=O)CCCC2)=O)CCCC12CCC2 C1(C(N2CC(C(=O)NC)C2)=O)CCCN(C(N)=O)C1.C12CCN(C1)C2=O c1(N2CCC(NC(CCn3cc(COCC)nn3)=O)C2)ccc(Br)cc1 C1(NC(c2c(COC)ncs2)=O)CCC(N(C(=O)CC2CN(C)CCO2)C)CC1 C(=O)(CC(O)CC(C)(C)C)N1CC(CN2CC(O)(C(C(=O)OC)F)C2)OCC1 CCCCCCC(C)C(=O)N1CC(C(=O)Nc2cc(C)c(O)c(C)c2)C(F)(F)C1 Cc1cc(F)cc(C(=O)NCCCCN(C(=O)Cc2nncn2C(C)C)C)c1C c1(NCC2CCN(C)CC2)[nH]c(=NCC(C)(C)C23CCC2(C)C3)nc2c1ncn2C C1(c2n(CC)nnn2)(NC2CC(CC3CC3)C2(C)C)CCS(=O)(=O)CC1 c1(CC)nnc(C)cc1C(=O)NCC12CC(CN1C(C1(C#N)CCOC1)=O)C2 C1(C(=O)NC(C=C)C2CCC2)C(O)CCN1C(=O)C(C1CC1)OCC N1(C(COCC(=C)C)=O)CCOC(CN(C)C(C2CCC2(F)F)=O)C1 C=C1CC(C(=O)OC)N(C(C2CCN(Cc3ccc(C)s3)CC2)=O)C1 C1(C(=O)NCc2cn(CC=C)nn2)CC12CCN(C(c1ccc(CF)cc1)=O)C2 N1(C(C2C(C)C2C)=O)CCC(C2(NC(=O)Cc3nncs3)CC2)CC1 n1(CC)ncc2c(NC3CC(NC(C4CCC5CC(C)CN5C4)=O)C3)ncnc12 n1(CCOC)cc(NC(c2conc2CNC(C2CCC(O)C2)=O)=O)cn1 C1(CNC(CSCCC)=O)CCC2CN(C(C3CC(C)(O)C3)=O)CC12 C1(N(C(c2ccn(CCC)n2)=O)C)CN(C(c2cn(CCO)nn2)=O)CC1F C1(C(N2CC(NC(CC3C(C)(C)COCC3)=O)(CO)C2)=O)CNC(=O)CC1(C)C C1(NC(c2cnc(CC)o2)=O)CCN(C(c2cccc(SC(C)C)c2)=O)CC1C N1(C(c2nc(N(C)C)sc2)=O)CCCC(NC(c2ccnc(S)c2)=O)C1 c1(CC(=O)OC)occ(C)c1C(=O)NCCN(C(=O)Cc1nonc1C)C(C)C C1(C(N)=O)Cc2cccc(NC(=O)C(c3cc(Br)ccc3Cl)N)c2C1 N1(C(CC2CC3(CN(C(c4cc[nH]n4)=O)C3)C2)=O)CC2CCCCCCC12 Cc1cc(C(N2CCC(NC(c3cc4c([nH]3)CCC4)=O)C2C)=O)cnc1C(F)F CN1CC(C)(C)CC1C(=O)NC1CC(CNC(=O)CCC2CC2(Cl)Cl)C1 c1(NCC(CNC(C(C)CSC(F)(F)F)=O)O)ncnc2ccc([N+](=O)[O-])cc12 C1(C(N(C)CCc2cccc(C#N)c2)=O)CCCCC1(C)C C12(C(=O)NCC3(C4CCN(C(=O)C=Cc5cocn5)CC4)CC3)CCC(CC1O)C2 C1(N(C(=O)CCNC(=O)Nc2ccccn2)CC)CCCN(C(=O)CCC(C)C)C1 c1(CC(=O)OC)ccc(OC)c(OC)c1Cl.c12ccc(ccc1=O)cc2 N1(C(C(C)=C2CC2)=O)CCC(C(F)(F)F)C(CNC(C2(C)CCC(=O)CC2)=O)C1 N1(C(C(C(C)C)F)=O)CCCCC(C2CN(C(C3CC(=O)C34CCCC4)=O)C2)C1 CC1CCc2[nH]c(=NCC3C4COCC34)[nH]c(=NCCCCCCCCO)c2C1 C1(CNC(CSc2c(C)n[nH]c2C)=O)CN(C(=O)C=CCN(C)C)CCC1(F)F c1(CC(N2CC(NC(c3coc(CC4CC4)c3)=O)C2)=O)csc2ccccc12 C1(NC(CC(CC)C)=O)CCN(Cc2ccc(N3CCOCC3)cc2)CC1(C)C N1(C(Cc2c(C)con2)=O)CCN(C(=O)C(c2c(C)noc2C)C)C(CO)C1 c1(C(=O)NCCC2N(C(COC(CC)CC)=O)CCCC2)ccnc(F)c1OC c1(OCC)ccccc1N(C(c1scnc1Br)C(=O)NC)C C1(C(=O)NCc2ccc(C)s2)CC12CCN(C(=O)Cc1cnn(C)c1C)C2 N1(C2C(C)SCC2)CCC(O)(C(N2CC(C(c3ccccc3)=O)C2)=O)CC1 CCCCCC(CC)C(=O)N1CCCC(F)(CNC(c2cnncc2O)=O)C1 C1(C(N(C2CC2)CC2N(C(CC3CC(CC)C3)=O)CCC2)=O)CCC(F)(F)C1O c1(OCC(=O)NCCC(C)NC(C(CC)n2ccnc2)=O)ccccc1C(F)F c1(C(=O)NC(CNC(CCN(C(CCC)C)C)=O)CO)ccnc(OC(C)CC)c1 N1(C(C2(OCC)CC2)=O)CCCN(C(c2[nH]nnc2C(F)F)=O)CC1 c1(C(N(CCC(C(C)C)NC(CC(C=C)CC)=O)C)=O)cc2cnn(C)c2s1 c1(CS(N2CC3CCN(Cc4ccccn4)C3C2)(=O)=O)c(F)ccc(F)c1F c1(C(=O)NC2CC(C)N(CCn3cccn3)CC2)coc2ccccc12 CC(C)(CC(=O)NCC(CC(F)(F)F)NC(=O)C1CCc2nccn21)C(F)(F)F N1(C(c2c(C)onc2)=O)CCC(C)C(NC(c2cc3sccc3s2)=O)C1C c1(CC(N2CC(CCNC(C(C3CCOC3)OC)=O)C2)=O)ccccc1C CN1CCN(C(c2cnsn2)=O)C(CNC(C2(Cc3ccccc3)CCC2)=O)C1 O(NC(=O)CC(C(F)(F)F)NC(=O)C(CC(CC)CC)CC)CC1CC(=C)C1 N1(C(CN2CCC(=O)NC2=O)=O)CC(NC(c2occ3c2CCC3)=O)CC2(CC2)C1 Cc1nn(C)c(F)c1C(=O)NCC1CCCC(NC(C2(C3CC3)CCCO2)=O)C1 C1(NC(C2NC(=O)OC2)=O)CCCCCC1C(=O)NCCn1cnnc1 c1(CC(=O)N(C(CCNC(COCCCOC)=O)C)C)ccnc(F)c1 N1(CC)CCOC(C(N2CCC(C)C2CNC(c2cccn2C(C)C)=O)=O)C1 c1(C(N2C(CNC(C3CSCC(=O)N3)=O)CC(OC)C2)=O)coc2c1COC2 c1(C(=O)NCC2CC(NC(=O)CCCF)C2)ccc(S(=O)(=O)NCC2CC2)o1 C=CCCCC(C(=O)NC1CC(CC(=O)OC)C1)NC(c1ccc(F)cc1)=O C1(CNC(C2CCC(OC)C2)=O)CCC2CN(C(=O)COC3CC(F)(F)C3)CC12 N1(C(=O)CO)CCC(C)(CCNC(=O)COC(c2c(COC)scc2)=O)C1 c1(C(=O)NC(C(=O)NC(CC=C)CC)Cn2cccn2)ccnnc1C C1(NC(Cc2c(C(C)(C)C)cccc2)=O)CN(C(C2CCOC2=O)=O)C(C)(C)C1 N1(C(CCC=C=C)=O)CCN(C(=O)CC2CCCC2C)C(C(C)(C)C)C1 CC(CCO)C(=O)NC(C1CCN(C(=O)CNC(c2cccs2)=O)CC1)C c1(C(N2CCC(N(C)C(C3CCCS3)=O)CC2)=O)ccc([N+](=O)[O-])cn1 C(=O)(CCC(F)(F)F)NCCOCCCNC(C1CC1C1CC1)=O N1(C(c2nc(C3CC3)cs2)=O)CC2CC1CN2Cc1nncs1 N1(C(c2ccc(C(C)C)s2)=O)CCN(C(=O)CC2(O)CCC2)C(C)C1 N#Cc1cc([N+](=O)[O-])ccc1NCCC1CCN(C(=O)CCS(N)(=O)=O)C1 C1(c2cn(CCCCC)nn2)CCN(C(=O)COC(c2ccccc2)(CC)CO)C12CC2 C1(C(=O)Nc2ccc(O)nc2)CN(C(c2ccc(Cl)cc2I)=O)CCC1O c1(C(=O)NCCN(CC(C)O)C(C2C(CC)(CC)C2)=O)ccc(NC2CC2)cc1 N1(CC(C)C)CC(C(=O)NCC2(NC(C3CNC(=O)N3)=O)CCC2)CC1=O CC1C(NC(=O)C2=COCCC2)CC2CCC1N2C(=O)CCCc1csc(=N)[nH]1 CN1CCC2C(CCCN2S(=O)(=O)c2scnc2C(=O)O)C1 CCC(CC)(CC)C(=O)NC1CC(NC(C2CC(O)CN2C(C)=O)=O)C(O)C1 N1(C(C(CC)CN(C)C)=O)CC2CCN(C(=O)C=C(C)Cl)CC2C1 c1(C(=O)NC23CC(C(N4CCC(F)(F)C(O)C4)=O)(C2)C3)ccc(Cl)c(Cl)c1Cl c1(OC)ccc2cc(C(N3CC4CC3(CNC(=O)C(F)OC)C4)=O)nnc2c1 c1(OC)cnc(Cl)c(C(=O)OC(C)(C)C)c1.C12CCC(C)(CC1)NC2=O c1(C(C(=O)NC2(CO)CN(C(C3N(C(C)=O)CSC3)=O)C2)C)c(C)nn(C)c1C c1(C(=O)NCCC(C)NC(C2=C(C)OCC2)=O)nnn2c1CCCCC2 C1(SC)CCN(C(C)(C)C)C1=O.C1(C2CC2)CC(C)N1 N1CCCCC1C.c1(C(C(=O)N(CC(CNC)O)C)(C)C)ccc(O)cc1 c1(OC)ccc(C)c(CCNCC2(c3ccccc3)CC(O)C2)c1 CC1=C(C(=O)N2CCC(N(C(=O)CCc3cnc[nH]3)CC3CC3)C2)CC1 CCCCCC(=O)NC12CC(C(N(C)C[Si](C)(C)C)=O)(C1)C2 C1(CNC(c2cnc(NC)s2)=O)CN(C(C2CC(O)CN2C(C)=O)=O)CC12CC2 N1(C(CC(=C=C)C)=O)CC(CNC(c2cc(F)cc(N)c2F)=O)C2(CCC2)C1 C1(C(=O)NCCC(C)N(C(c2cnc(OC)c(C)c2)=O)C)CC2(C1)CC(C)(C)C2 C(=O)(C1=NN(CC(C)C)C(=O)CC1)NCC(CC)NC(c1cc(CCC)on1)=O CCC(C)(C)CCNC(=O)C(Cc1cn[nH]c1)NC(=O)CC1CNC(=O)O1 C1(C(N(C(C)CC2CC2)C)=O)CN(C(C2CNC(=O)N2)=O)C(C)(C)C1 C(=O)(C(CNC(c1ncnc(C)c1C)=O)C(C)(C)C)NC1(CC(=O)OC)CC1 Cc1cnc(C(=O)N(C)CC2CCN(C(c3ccc(C(C)F)cc3)=O)C2)nc1 c1(C(=O)OC(C)C(C)(C)C)ncccc1CCNC(=O)OC(C)(C)C N1(C(C2C(C)CC(C)O2)=O)CCN(C(=O)CCN2CCCCC2=O)C2(CCC2)C1 C(C(C)CC(=O)NC(C(N)=O)C1CC1)NC(C1(CCC)CC(=O)C1)=O CC1CN(C(=O)C(N)=O)CCC1NC(C1(C)CN(C(=O)OC(C)(C)C)C1)=O c1(C(c2n(C(CNCC3CCCCC3)C)nnn2)OC)sccc1S(N)(=O)=O N1(CC)Cc2cc(CN3CCCCC3c3cccc4ccccc34)ccc2C1=O Cc1ccc(CNCC2CCCCN2S(=O)(=O)c2cn[nH]c2)cc1O C1(CNC(CC=C)=O)CN(C(=O)COC2CCC(C)CC2)CC1C C1(C(=O)NCCN(CC(C)O)C(c2cc(C3CCC3)n[nH]2)=O)(OC)CC(C)C1 Cc1cccc2c(CCC(N3CCC(CNC(C4C(C)C4C)=O)C3)=O)c[nH]c12 Cc1ncc(C(=O)NCC2CCCC2C(=O)NOCC(F)(F)F)c(=N)[nH]1 c1(C(N(CCCNC(C2CCSCC2)=O)CC)=O)ccn(C(C)C)c1C c1(OC)ccc(COC(c2ccccc2C(C)=O)=O)cc1F C1(C(N(C(CC)C(=O)N(C)CC2(O)CCC2)C)=O)CC2C(C1)C2(C)C N1(C(c2c(C)scn2)=O)CCC(C)(CC(=O)NCC2(C)CC3(CC3)C2)C1 c1(NC)ccc(Cl)c(C(=O)NC2CC(C)N(C(c3cn(C)c(O)n3)=O)C2)c1 N1(C(C(CC)n2ccnc2)=O)CC2CC1(c1cn(CC3CCOC3)nn1)C2 c1(C(=O)NCC)cccc(C2CC2)c1C.c12ccc(nn1)N1CCN(CC1)C2.NCC c1(CCCC=C)ccc(C(=O)NCC2CN(C(C3CCCCS3)=O)CC2C)cc1 N1(C(C2CCN(C(CCC)C)CC2)C(=O)NC2CC2)CCC2(C1)NC(=O)N(C)C2=O CCC(CO)C(=O)NCCC1CCCN(C(c2cccc(C(C)(C)C)c2)=O)C1 C(=O)(C(F)C(C)C(F)(F)F)NC(c1cn(C(C)CNC(=O)N(C)C)nn1)(C)C c1(C(C(=O)N2CC(C3(C)N=N3)C2)NC(=O)OC(C)(C)C)ccccc1 c1(CC(=O)N(C(C(=O)N2CC(C(=O)NC)C2)CC)C)c(C)noc1C N1(c2nc(C)c(Br)cn2)CCC2(CCN(C(=O)C(C)(C)CO)C2)C1 n1(CC(=O)NC2CCC(NC(CC(=C=C)C)=O)C2)c(=O)nc(O)c2ccccc12 N1(C(c2ncc(C)cn2)=O)CCC2(CCCN(C(=O)CC3CSC3)C2)CC1 n1(CC)ncc(C(=O)NC2COCCC2NC(=O)CN2CC(C)C2)c1Br Cc1cc(C(N2CCC(CNC(C3CCOC3)=O)CC2)=O)nn1CCO c1(C(=O)NC2C3CN(C(c4nc(CC)sc4)=O)C2C3)cccc2c1OCC2 c1(C(N2CCC(CN(C(CCC(=C)Cl)=O)C)C2)=O)nccc(N)c1Cl c1(C(N(CC(C)NC(c2cc(C)nn2C)=O)C)=O)ccc(Cl)c(F)c1F N1(C(C(C)(C(C)C)n2cc(CC(=O)OC)nn2)=O)C2CCCC(O)C1CC2 c1(NCCC2(NC(C(C)Oc3ccccc3Cl)=O)CCC2)nc2ccccc2o1 c1(N2CCC(CC=C)(NC(C3CC(F)(CO)C3)=O)C2)ncnc(Cl)c1CC C12(NC(C(C)c3ccco3)=O)CCCN(C(c3cc(Cl)ncc3Cl)=O)CC1C2 C1(NC(C(CC)OCC)=O)CC(C(=O)NCCCOC(F)(F)F)=CC1O n1(CCCC)cc(C(=O)NCC(C)NC(=O)CCNC(N)=O)c(C)n1 c1(C(=O)NC2CN(C(CNC(CC)=O)=O)CC2C)ccc(C(C)(C)C)cc1C N1(C(c2c(NS(C)(=O)=O)cc(Br)cc2)=O)CCC2(CCC(C(=O)O)NC2)CC1 C=C(C)C1OCCC1C(N1CC(C(O)C(=O)NCCN2CCCC2=O)C1)=O CCCCC(C(=O)N1CC(O)CC1CNC(c1n[nH]cc1C1CCC1)=O)C(C)C C(C(C(C)C)NC(C1(OCC)CCOC1)=O)NC(CC1CC(=C)C1)=O N1(C(COC2(C#C)COC2)=O)CC2(CC(NC(c3csc(O)n3)=O)CO2)C1 C12(NC(c3n(CCC)ccc3)=O)CCC(CC1)N(C(c1ccc(CSC)o1)=O)C2 C1(NC(c2c[nH]c3nccc-3c2)=O)CC2CC1CN(C(c1ncc[nH]c1=O)=O)C2 c1(CN2CC3C(C(=O)NCc4ccc(C)nc4)(C3)C2)[nH]nc2ncccc12 CC1(C)C(CN)CCS1(=O)=NC(=O)NS(=O)(=O)N1CCCC1 CCC(C#N)C(=O)N1C(CNC(=O)CSc2nncn2C)CC2CC12 C1(COC)CN(C(=O)C(C)(C)c2ccno2)CCN1C(=O)CC1CC1(Cl)Cl CCCC(CCCNC(=O)C(COC)N(C)C)NC(=O)C=Cc1cnc(C)s1 O=C(CC(O)CNC(c1ccc[n+]([O-])c1)=O)Nc1ccccc1C1CC1 C1(C(=O)NCCOCC(=O)NC(C(=O)NC)C2CC2)CCCN(C)C1 CC(=O)CCCCC(=O)N1CCC2CN(C(=O)C(C)Cn3cccn3)CC12 C1(C(N2CC(CCNC(c3cnc(C(C)=O)s3)=O)C2)=O)CC2C=CC1C2 Cc1ccc(NC(C2CC(O)CN2CC2CC3(CCC3)C2)=O)c(-c2cnco2)c1 c1(OC)ncc(Cl)cc1C(=O)NC1CN(C(c2cncc(Br)c2)=O)CC1(F)F N1(C(C(C=C)(C)C)=O)CC(NC(c2cccc(Br)c2Cl)=O)CC(F)(F)C1 N1(C(Cc2cn(C)nc2)=O)CC(NC(=O)C(C)(C)c2ccnn2C)CC(O)C1 Cn1nnc(C(N2CCC(C(C)(C)C(=O)NCCc3csnn3)C2)=O)c1N CC1CC=C(C(=O)NCC2(CNC(c3cccn4nnnc34)=O)CC2)CC1 CC(C(=O)NNC(=S)Nc1ccc(Cl)cc1)N.C12(CN)CCCC1C2 C1(CNC(c2ccc(CC)cn2)=O)CCC2(CN(C(C3CCC(C)(C)O3)=O)C2)O1 N1(C(c2scc(C)c2)=O)CCCC(C2CCN(C(C3(C4(O)CCC4)CC3)=O)C2)C1 C1(CNC(c2c(C)nc[nH]2)=O)CCN(C(=O)C=CC2COC(C)(C)O2)CC1(F)F CC1CN(C(=O)COC2(C)CN(C(c3cc(C#N)c[nH]3)=O)C2)CC(C)(C)C1 C(=O)(C(C(=O)NC(CNC(c1sccc1C(C)C)=O)C(C)(C)C)C1CC1)OCC CC1=C(C(=O)N2CCCC2C(C)(C)NC(C2(C)CCC2)=O)CCS1(=O)=O c1(C(=O)NC2C3N(C(c4c(NC)cnnc4)=O)C(CC3)C2)ccc(F)c(F)c1F C1(C(N2CCC2C2CCOCC2)=O)(NC(C(C2CN(C(N)=O)C2)O)=O)CCSC1 S(=O)(=O)(c1cnn(C)c1)NC12CC(C(=O)Nc3c(C(C)=O)cc(F)cc3)(C1)C2 Cc1cc(C(=O)NC2CN(C(C3CCCCS3)=O)CC2O)c2cnccc2c1 C(=O)(C1=COCC1)NC(CN(C(c1nc(Cl)cs1)=O)CC)C c1(-n2cc(C(C)NC(C(=O)N(CC)CC)C)nn2)ccc(Cl)cc1Cl CS(=O)(=O)CCC(C(N)=O)NC(c1ccccc1-n1cccn1)=O N1(C(CC(=O)OC(C)(C)C)=O)CC2CC(C(=O)NCCc3cccc(F)n3)(C2)C1 N#Cc1c[nH]c(C(=O)NCC(CO)NC(=O)Cn2nnc(C(F)(F)F)n2)c1 Cc1nn(CCN2CCN(CC(C)C)C(=O)C2)c(C)c1C n1(CC(=O)Nc2ccc(Oc3ccc(OC)cc3)nc2)ncc2ccccc12 c1(C(=O)Nc2cccc(Br)c2)ncn2cc(-c3cccc(OCC(F)F)c3)sc12 c1(C(N(CC)CC2CCCCN2C(C2CCN2C)=O)=O)ccc(C#N)cc1 C1(CCC)(NC(c2cccc(C)c2C)=O)CCCN(C(=O)COCCCOC)C1 C(=O)(C=CSc1nc[nH]n1)N(CCC)CCNC(c1cnc(C(C)OCC)s1)=O c1(C(=O)NCC2(C)CCN(CCC=CCC)CC2)cc(C)nc2onc(C)c12 C(C)(C(C(=O)NCCN(C(C1(c2ccccc2)CC(O)C1)=O)C1CC1)N(C)C)OC N1(CC)C(=O)CCC1CC(=O)NC1(C)CN(C(C2(CO)CC2)=O)C1 n1(CC(=O)NC2CCCN(C(c3cnc(Cl)c(Br)c3)=O)C2)nnc2ccccc12 c1(OC)cc(C(N2CCCC2c2c(Cl)cccc2Cl)=O)cn2c(Br)cnc12 N1(C(CC(C)(F)F)=O)CCOCC(CNC(C23CCCCC2C3)=O)C1 CC(CN=C(NNCC1CC1)NCC(C)(Cc1ccccc1)CO)CC(F)(F)F N1(C(C2CCN(C(C(CCC)C(C)C)=O)CC2O)=O)CCCC2C1CCN2C c1(C(N2CC(C)(N(C(=O)CNC(N)=O)C)C2)=O)ccc(-n2cccn2)nc1 N1(C(c2noc(C)c2[N+](=O)[O-])=O)CCC2(CCCN2C(C23COCC2C3)=O)CC1 CC1CN(C(C2(S(N)(=O)=O)CC2)=O)CC1NC(c1coc(C2CCOCC2)n1)=O c1(C(=O)NC(CC)(C)CNC(C2(COC)CC2)=O)cnn2ccnc(C)c12 N1(C(C2C(SC)CCC2)=O)CC2CC(C1)C2NC(C1CC2CC2C1)=O c1(CN(C(C)C)CCN(C(C)C(=O)NC2CCC(C)CC2)C)ccc(F)cc1F C(CCCCCNC(=O)CC1CC12CC2)N(C(=O)Cc1cncn1C)C CCC(C#N)(CC)C(=O)NC1CC2CC(NC(=O)CNC(=O)CCC(C)C)C1C2 c1(C(=O)NCC(C(C)(C)C)NC(C(C)SC(F)(F)F)=O)ccc(N)c(Cl)c1 N1(C(CCN(CCC)C)=O)C2CCC1CC(NC(=O)C(F)(F)CC)C2 C#Cc1cccc(C(N2CCCC(NC(=O)CC3CCC(=O)NC3=O)C2)=O)c1F c1(C(=O)NC(CCN(C(C2(COC)CC=CC2)=O)C)C)cc(OC(F)F)n(C)n1 N1(C(CCCNC(C)=O)=O)CCC2(CC1)CC2NC(=O)C(F)(F)CC1CC1 CCCC(C)CCNC(c1ccc(CNC(c2c[nH]c(=NC)s2)=O)o1)=O C1(NC(c2nc(C(=O)OCC)sc2)=O)CN(C(c2coc(Cl)n2)=O)CC2CC12 n1(C(C)C)ccnc1C(=O)NCc1ccc(C(=O)NCC2CCC(O)C2)s1 c1(NC(C(C)(N(C(CC=CCC)=O)C)C2CC2)=O)ccn2nccc2c1 CCCC(CNC(=O)CCC1OCCO1)C(=O)NCCC1CCC(C)CC1 Cc1cc(I)ccc1C(=O)NC1CCC(C(=O)Nc2nc(Br)cn2C)C1 c1(C(=O)NC2CCN(C(C3CC(=O)OC3)=O)C2)nc(Br)[nH]c1C(F)(F)F N1(C(c2c(Cl)c(C)n(C)n2)=O)CCC(NC(C2OCCO2)=O)C(C)(C)C1 CCCC(C)CCCC(=O)N(C)C.N12CC(O)CC1Cn1cc(nn1)CCC2 N1(C(C2(C#N)CCC2)=O)CC2CCC2(CCNC(C2(F)CC2)=O)C1 c1(CC)ccc(C(=O)NCCOCCCNC(C2CCCC(C)CC2)=O)cc1N O=C(C1CCc2cccnc21)N1CC2CCC(C1CO)N2C(=O)COCCF c1(C(N(CCOC)CCNC(c2cccn2C)=O)=O)nc(C)ccc1F C12CC=CCN1C2=O.C1(C2CC2)CCCN1C(=O)CC1(N(C)C)CC1.CO C(C)(C)(CCNC(=O)C=CSC)NC(C1(COC)COC1)=O c1(NC)ccc(F)cc1C(=O)NC1CCC(NC(c2cc(C)ncc2C)=O)CC1 C12(C(=O)NCC3CCCCN(C(C(C)SC(C)C)=O)C3)CCCCC(F)(C1)C2 c1(CN2CCCC(O)(C(C(=O)NC)(F)F)C2)nc(C)c(Cl)cc1Cl c1(C(N(CCCN(C)C(c2cnn(C)c2)=O)C)=O)cccc(S(C)=O)c1 C(=O)(C(F)CCC(C)C)N1CC(COC)N(C(=O)C(C)N(C)C(C)=O)CC1 c1(C(=O)NCC(CO)NC(=O)COCC2CCCOC2)c(O)nnc2c1CCC2 C(=O)(C(O)CCCCC)NC(C(=O)NC(CC=C)(C)C(F)F)C CC(CCc1cnn(C)c1)N=c1[nH]n2ccnc2s1 Cn1nc(C2CCCN2C(c2cc3cc(Br)cn3cn2)=O)c2ccccc2c1=O c1(C(N2C(C)C(NC(=O)C(O)C3CCCC3)CC2)=O)cn(C)c(=O)cn1 c1(C(=O)NCC(CNC(C2CCC(C(=O)OC)C2)=O)O)nccn2cc(C)nc12 N1(C(C(CCC)N(C)C)=O)CC(C)(C)OCC1CNC(c1cc2[nH]ccc2s1)=O CCC(C(=O)NC(C)(CNC(c1c(OC)ccc(Cl)c1F)=O)CC)C(F)(F)F O=C(CCCc1nccs1)NCC(CNC(c1cc(Br)c[nH]1)=O)CO C1(C#N)(C(N(CCOCCN(C)C(c2cncs2)=O)C)=O)CCCCC1 C(CCC(=O)NCC1CC1NC(=O)CCCc1cc(C)no1)NC(=O)NCC#C N1(C(=O)NCC(=O)NC(C2(Sc3ccncc3)CC2)C)CC2CC3CC2C1C3O C1(CNC(C(C=CC)O)=O)CN(C(C2CC2c2ccccc2)=O)CC12CCC2 C#CCC(C(=O)NCC1CCN1C(C)(C)C)NC(c1cnn(C)c1Cl)=O c1(C(=O)NCCOCCNC(Cc2c(C)nccc2)=O)cnn2cccnc12 N12C(=O)CCN(C1=O)CCCCC2.N1(C(C)CN(CC(F)(F)F)C)CCCCC1 C(=O)(C1=CCCCO1)NCc1ccc(C(N2C(C(CCC)C)CCC2)=O)s1 Cc1ccncc1C1CC1C(=O)N(C)CC1CN(C(=O)C(C)C)CCO1 C#CCC(O)C(=O)NC1(CO)CN(C(c2cccc(-c3cscn3)c2)=O)C1 c1(NC2CN(C(c3cc(C)[nH]c3)=O)CC2C)ncc([N+](=O)[O-])cc1Br c1(OCC(=O)NCC)cccc(NC(=O)CN2CCOC(CC(N)=O)C2)c1 c1(C(c2n(CCCSCC)nnn2)NCC(C(C)C)OC)cccc(C)c1F C1(NC(C2(COC)CC2(F)F)=O)CCN(C(C2CSCN2C)=O)CCC1CO C1(CCNC(c2cc(Br)ccn2)=O)CCN(C(CC2C(CC)C2)=O)CC1 O=C1CC(C(N2CCCCC(CNC(=O)CCOC3CC3)C2)=O)C2(CCC2)C1 N12CCCC1NC(=O)COCC2=O.C1(CCOCCOCCOC)CCCO1 Cc1ccc2c(C(=O)NCCC3COCCN3C(=O)CCC(N)=O)onc2c1 c1(C(N2CC(OCCC(=O)N(C)CCn3cccn3)C2)=O)ccncc1N(C)C C1(NC(C(C)NS(CC)(=O)=O)=O)CN(C(=O)C#CC2CC2)CC1C(F)(F)F N1(C(c2c(-c3cn(C)nc3)[nH]cc2)=O)CC2CC(C1)CN(C(=O)C(O)C1CC1)C2 N1(C(c2ccn(C)n2)=O)CCC(C2CC2)C1CNC(C1CS(=O)(=O)CC(=O)N1)=O c1(CN(C2COCCN(C)C2)CC2CN(C)CCO2)nn(C)c2c1CCC2 c1(C(N(CCCNC(=O)C(c2cccs2)SC)CC)=O)nccc(Cl)c1C C1(O)(CCNC(C2CCCCCCC2)=O)CCN(C(C2CC2C(F)F)=O)CC1 C(C(CC(C)C)C(=O)NCCCCC(=O)NOCC1CCOC1)OC C1(C)(C(N2CCC(NC(c3ccc(C)nn3)=O)C2)=O)CC(C(C)(C)C)=NO1 c1(CC)cc(Cl)ccc1C(=O)NCc1nc(CNC(=O)C(C)CC2CC2)cs1 c1(OC)cc(Cl)c(C)cc1C(=O)OCc1cn(-c2c(C)cccc2C)nn1 C=CC1(C(=O)NCC2(O)CCCC2(C)C)CCN(C(=O)C2=CCN(C)C2)CC1 CC(CCC(=O)NCCC1(CNC(C2CCCN2C)=O)CC1)N(C)C C(C(CO)(CO)NC(C1CC1F)=O)N(C(c1ccn(COC)n1)=O)C n1(CC)nnc2c1C(C(=O)N1CC3OCC(C)C3C1)CN(C(=O)C=CC1CC1)C2 N1(C(CCC=CC)=O)CC(NC(=O)C=CCOCCOC)CC2(CC2)C1 c1(CC)nc(Cl)c(F)c(=NC(CNC(=O)CCSC)CC)[nH]1 C12(NC(=O)NC3(c4ccc(F)c(F)c4)CCC3)CCCCCC1OCC2 N1(C(C2(C)CCC(C)C2)=O)CC2CN(C(c3cc(C(F)(F)F)ncn3)=O)CC2C1 c1(C(N2CC3CC3C2)=O)cnn2ccc(-c3ccc4cncn4c3)cc12 C1(Cl)(C(=O)NCC2CCN(C(c3ccn(C(C)(C)C)n3)=O)C2)CC12CCC2 CCC(CN(C)C)CC(=O)N(C1CCN(C(=O)Cc2c(Cl)cnn2C)C1)C C1(C(=O)NCCCC2N(C(C(c3n(C)ccc3)=O)=O)CCC2)CC(F)C(=O)N1 c1(N2CCCC(CCC)C2)nc(N(CC(C)C)C)nc2c1CCCC2 c1(C(=O)NCC(CNC(C(C)n2cccn2)=O)(C)O)c(Cl)ccc2c[nH]nc12 C1(c2cc(OC)c(O)c(F)c2)CCCN1N1CCCC1CCF N1(C(C(CSC)OC)=O)CC(CN(C(=O)Cc2cccc(C)c2)C)C(C)(C)C1 c1(C(=O)NCCC(C)NC(=O)Cc2ccccc2Cl)ccc(C(=O)N(C)C)cc1 n1(CC)c(C)nn(CC(=O)NCCC2CCCN2C(=O)CCC(C)N(C)C)c1=O c1(C(N2CC(N(C(C)=O)C)C(F)C2)=O)n[nH]c2cccnc12 C1(NC(Cn2nc(C)oc2=O)=O)C2CC3C1C3C2C(=O)NCCC1CCCCO1 C(=O)(CC1NC(=O)c2ccccc21)NCCCNC(=O)CC1CCC(F)(F)CC1 c1(CN2C(C)(C(N3CCN(C4CC4)CC3)=O)CC2)c[nH]c2cc(F)c(F)cc12 c1(CC(=O)NCC2C(NC(C3(C)N(C)CCC3)=O)CCC2)cncc2ccccc12 Cc1csc2cc(C(N3CC(NC(=O)CCC4(C)CC4)C4CC4C3)=O)[nH]c12 C1(OC)CC(CNC(C2(CO)CCC2)=O)N(C(=O)Cn2cc(Br)cn2)C1 N=c1ccc(C(=O)NC(C(=O)NCCN2CCCOCC2)C2CCC2)c[nH]1 N1(C(C(CO)NC(=O)NCCO)=O)CCC(COc2ccccc2)CC1 C(=O)(C1=CCCC1(C)C)NC(CN(C(C1Cc2nnsc2S1)=O)CC)C CC(C)C(C)C(CNC(C12CCC(CC1)O2)=O)NC(c1cc(=O)n(C)cn1)=O C=C=CCC(=O)NC1CCOC1C(=O)NC(c1ccns1)C CCCC(CCC)CC(=O)N1CCC(CO)C(NC(=O)CSCCC(C)C)C1 C(=O)(CS(=O)(=O)C1CC1)NC1C(C)(C)CN(C(c2ccc(N)c(O)c2)=O)C1 c1(C(=O)NC(C(=O)NCC)C)ccc2c(n1)CN(C(c1cnncc1C)=O)CC2 C1(C(N2CC(C)C(C(=O)NCCN3CC=CCC3)C2)=O)CCCC(C)(C)C1 C(=O)(C(C)C(O)CC(C)C)NCC1=CCN(C(c2c(C)c(Cl)cnc2)=O)CC1 c1(Nc2cc(OCC)ncn2)ccc2c3c(cccc13)CC2 c1(-c2cccc(OC)c2F)ccc(S(=O)(=O)N2CCN(CC(F)F)CC2)cc1 c1(-n2c(C3C(C)=CCS3)nc(-c3ccc(C4CCC4)cc3)n2)cc(C)ccc1C c1(C(N2C(C)CN(C)CC2)=O)cc(O)nc2c1CN(C(=O)CSCC(N)=O)CC2 c1(C(N(CCCC(C)O)C)=O)cc(-c2cn(CCC(C)(C)C)nn2)cnc1O CCCCC(F)C(=O)NC1CC2CC(NC(c3cccc(C)c3Cl)=O)C1C2 N1(C(c2c(NC)nccc2)=O)CCC(C)C(NC(c2coc3c2COC3)=O)C1C C1(OC)CN(C(c2cc(-c3cnn(C)c3)[nH]n2)=O)CC1NC(=O)C(C)(C)F CCCCCC(O)CC(=O)N1CC2CCCC2(NC(=O)CC2CNC(=O)O2)C1 Cc1[nH]c(C(=O)N(CCO)CCO)c(C)c1C(=O)Nc1nc(Cl)cnc1Br C1(CNC(C2(C)CC(=C)C2)=O)N(C(=O)CC2CNC(=O)C2)CCCC1(C)C c1(CCCC)nc(C(=O)NC(C)C(C)NC(=O)C(=O)N(C)C)cs1 c1(OC)ccc(CCCC(N2CCOC(c3ccc(Br)cc3)C2)=O)c(Cl)c1 N1(C(CCN(C(=O)C=CCN(C(C)C)CCN(C)C)C)=O)CC2CCC1C(O)C2 Cc1ccnc(C(=O)NC2CCC2CNC(c2cnc(O)n2C)=O)n1 Cc1ccc(NC(C2(C)CCN(C(=O)Cn3ccnc3)C2)=O)c(Br)n1 C(CCC(C(=O)N(C)Cc1ccccn1)NC(=O)C(C)C1CCCC1)OC c1(NC(C)C)cnccc1NC1(CC2CC2(F)F)CCCCC1 CC(C)C(F)C(=O)N1CCC(COC2CCN(C(=O)C(C)n3cnnn3)C2)CC1 C1(O)(C(C)NC(CC(CC)C)=O)CCN(C(c2cnc3sccn23)=O)CC1 c1(C(=O)NCC2C(NC(C(N)=O)=O)CCC2)cc2ccc(Br)cc2cn1 c1(C(=O)NC(CNC(C(F)=CC)=O)(C)C2CCC2)ccnc2c(F)cccc12 Cc1nn(C)cc1C(N1CCC1CNC(=O)C(c1ccc(Br)cc1)C)=O CCC(CC(=O)N1CCOC(N(C)C)C1)N(C(=O)CCn1cncn1)C C1(C(=O)NC(C=CC(=O)NCC2(CC=C)CCCC2)C)CCCN(C)C1 C12(NC(=O)C=CC3CCOC3)CCCC(CN(C(=O)CC3CCC=CCC3)C1)C2 C=CCN=C(NCc1ccc(F)cc1C)NCC1CC(C)(c2ccccc2)C1 CCCC(CC)CCC(=O)NC(CN(C)C)C(=O)NCC(C)(C)C(N)=O C1(CNC(C=C(C)C)=O)CCN(C(c2cccc(-c3nnco3)c2)=O)C12CC2 N1(C(C(C(C)C)CN)=O)CCC2(CCC(O)C2)CC1 S(=O)(=O)(c1cnc(N2CC(C3CC3)OC(C)C2)c(Cl)c1)NCc1ncc(CC)s1 N1(C(C2(C)CCNC(=O)C2)=O)CCCC2(C1)CN(C(C1COC(=O)N1)=O)C2 c1(C(N2CC(C)CC(NC(c3c(CC)[nH]cc3)=O)C2)=O)c([N+](=O)[O-])c(C)nn1C N1(C(c2c(C)occ2)=O)CC(CC(=O)NCCN=[N+]=[N-])C(C)C1 C(CC(C(=O)NC12CC1CN(C)C2)NC(C1C(C)C1C)=O)=CC c1(C(=O)Nc2cccc(OCCOC)c2)cnc2ccccc2c1 C(=O)(C(C)(C1(C)CC1)OC)NCC(C)N(CC(=O)NCC#C)C(C)=O N1(CC23OCC(COCC)(C2)C3)CCCC(C)C1CO C1(N(C(=O)C2=COCC2)c2cc(CC)no2)CCC12CCNCC2 C(=O)(CCCC(=O)NC1CC(C)N(C(=O)C=CC2CCCN2C)C1)NCC N1(C(C=CCOC)=O)CC(F)CC1CN(C(=O)Cn1nnc(C)n1)C C1(C(=O)NCCC(C)NC(C2(C(F)(F)F)CCCC2)=O)CC=CCC1 c1(C(N2CCC3(C(N4CCC(C(C)O)C4)=O)C(C2)C3)=O)cnc2ccoc2c1 C1(C(=O)NC(C(c2ccc(Br)cc2)OC)C)CCC2(CCC2)C1 N1(C(CC(CC)OC)=O)CC(CNC(C2(C)CC3CC3C2)=O)C(F)(F)C1 C1(C(=O)NCC2(C)CCCN2C(c2cccc(N)c2)=O)CCCCC1(C)C c1(CN2C(C(=O)Nc3ccc(C(=O)OCC)cc3)CC2)cccc2ccoc12 N1(C(C2CC2Cl)=O)CC2(C(=O)NC(CO)C(F)(F)F)CCC1CC2 C(C(C)(O)CC(=O)NCCCNC(=O)C=CCN1CCCC1)OC N1(C(c2c(OCC)scc2)=O)CCC(OCCNC(c2cc(C#N)ns2)=O)CC1 c1(-c2ccn(CC)n2)cnc(NCc2ccc(OC)cc2F)c(O)c1 C(=O)(C1=C2CCCN=C2NN1)NC1C(C)N(C(C2CC3CCCC3C2)=O)CC1 C1(NC(C2CC(Cl)(Cl)C2)=O)CC2(C1)CC2NC(=O)C(O)CC1CC1 n1(CC(=O)NC2(C)CN(C(=O)C(c3ccccc3Cl)O)C2)cc(S(C)(=O)=O)cn1 C1(C(=O)NCCN(C(CC=CC=C)=O)CC2CC2)OCCC1C(F)(F)F c1(OC)ccc2c(C(=O)NCC(C)CNC(=O)CCCCC(N)=O)n[nH]c2c1 C1(N(C)C(C2(CO)CC(C)(C)C2)=O)CCN(C(=O)CCNC(=O)CO)CC1 C1(C(=O)OC)CN(C(C2CC2CNC(C2CCC2C)=O)=O)C(C)(C)C1 C=C=CC(C)C(=O)NC(C)(CSC)C(=O)NC(CC1CC1)C(=O)OC c1(C(=O)NCC(CN(CCC)C(C2CN(CC)C2)=O)(C)C)cnc(OC)c(C)n1 CC(C(=O)NCCN1CCN(C(c2ccn(CCN(C)C)n2)=O)CC1)C(F)F c1(C(=O)NCC(CC(=O)NC2CC(OC)C2)OC)cnc(O)c(F)c1 C1(NC(Cn2cc(C(=O)NC)nn2)=O)CN(C(=O)CN(C)CC)C2(CCOC2)C1 C(=O)(CC1=CCCCC1)NC1(C)CN(C(=O)CCCc2nc(C3CC3)no2)C1 c1(C(N(C(CNC(C(CC)=CC)=O)C2CC2)C)=O)cnc2c(c1)NC(=O)CN2C C1(NC(c2cc(C)ns2)=O)CN(C(=O)C(C)(C)c2ccnn2C)CC(C)(C)C1 N(C1CCC(NC(c2nncs2)=O)c2ccccc21)C(=O)CC12CCC(CC1)C2 C1(C(N(CCNC(=O)C(=Cc2cccnc2)F)C2CC2)=O)CCc2c[nH]nc2C1 C(c1ccc(Cl)cc1)=CC(=O)NCC1C2CN(C(=O)CCN3CCOCC3)CC12 C1(CCOC)CN(C(c2cscc2F)=O)CCN1C(C1CN(S(C)(=O)=O)C1)=O N1(C(Cc2c(C)ccnc2)=O)CC(NC(=O)CCOCC(F)F)CC12CCOC2 N1(C(C(C)(C(C)C)OC)=O)CCN(C(=O)C=Cc2ccccc2)CC(O)C1 CS(=O)CCC(O)C(=O)NCC1(NC(c2cnc(=N)[nH]c2)=O)CC1 N1(C(C(C)C(C)(C)C)=O)CC2(CCN(C(=O)CCF)CC2)CC1C n1(Cc2cn(C(C(N3CC(CC(=O)OC)C3)=O)C)nn2)cc(C(C)=O)nn1 C(CO)(C(F)(F)F)NC(CC=CCNC(CCOC)=O)=O c1(C(=O)NC2C(NC(CN(CC)CC)=O)CC2)nc(C)ccc1OC C12(CCNC(c3c(CC)nn(C)c3)=O)CCC1CN(C(=O)Cc1cncn1C)C2 N1(C(C2(C)CN(C(=O)C=C3CCC3)C2)=O)CCC2CCCCC2C1 n1(CC(C(=O)OCCSCCCCCC=C)(C)O)c(C)cccc1=O c1(C(=O)NCC(CC)(C)NC(=O)CC2CC(C)C2)cc(Br)c2nccn2c1 c1(C(=O)NC2CC(NC(c3c(C)cn(C)c3)=O)C2)nnc(O)cc1O C1(C(=O)NCC(CC)NC(c2cc(CCC)[nH]n2)=O)CCCC(C(=O)OC)C1 c1(C(N2CCN(C(C(CC(C)C)O)=O)CC2CF)=O)noc2c1CC(F)(F)CC2 CC1(C)CC(C(N2CC(CC(=O)Nc3ccccn3)C2)=O)N(C(=O)C2CC2)C1 c1(C(=O)NCC(CNC(C2ON=C(CC)C2)=O)(C)O)ccc(Cl)nc1OC1CCC1 C1(C(=O)NCC(C)N(C(=O)CC2(COC)CC2)CC)Cc2nnc(C)n2C1 C(=O)(CCCCN(C)C)NC(C1CCN(C(C2C(CCC)C2)=O)C1)C N1(C(=O)OC(C)(C)C)CCC2CN(CC=CCO)C2C1 C1(C(=O)NOCC2CCCC2)(CC=C)CCCN1C(=O)C(C)OCOC c1(C(C)Oc2cnccc2NC(c2nc(C(F)F)cs2)=O)cc(F)cc(C#N)c1 N1(C(C(CC)n2cncn2)=O)CCN(C(=O)CCN2CCC2)CC1CC c1(CCC(=O)NC2CCC(NC(=O)C=CC=C(Cl)Cl)CC2)nnc(O)nc1O C(=O)(C1=NOC(C)C1C)N1CC(CC(N2CC3C(CC)(C3)C2)=O)OCC1 CC(C)CC(CNC(C1(c2cc[nH]n2)CC1)=O)C(=O)NC1(C)CCCC1C C(=O)(C1CCCc2nc[nH]c21)N(CCCCCNC(C1CCS(=O)(=O)C1)=O)C Cc1nc(N(C)CC2CCN(C(c3ccc(C4CC4)cc3)=O)C2)c(F)c(C)n1 N1(C(C(n2ncc(C)c2)C)=O)CC2CC2C1C(=O)N(CC1CC1)CC1CC1 C(C)(C)(CCCC(=O)NC1CC12CCCCCC2)NC(C1CC=C(C)CC1)=O c1(C(N(CCNC(C2CC(=C)C2)=O)CCC)=O)cc2c(OC)cccc2[nH]1 c1(C(N2C(C(C)NC(C(C)OCC)=O)CCC2)=O)cc(F)c(F)cc1O CC1=C(C)CC(C(=O)NCC2C(C)CCCN2C(c2ccc(=O)oc2)=O)CC1 C1(NC(c2sccc2F)=O)CCOCC1C(=O)NCCCN1CCCC1=O C1(CNC(C=CC(C)C)=O)CCN(C(C2CCC3(CCC3)C2)=O)C1(C)C C12(NC(C=CCCC)=O)CC1CN(C(c1cccc(NS(N)(=O)=O)n1)=O)C2 CCCC(C)(O)CC(=O)NCC1CCN(C(=O)CCC2CCCO2)C(C)C1 c1(CCC(=O)N(C(CNC(=O)CC2CC3CC3C2)C2CC2)C)nccn1C(F)F N1(C(=O)Nc2c(-c3cc(C)sc3)nccc2)CCCC2(CCC2)C1 c1(CC2N(CC3(C(OC)OC)CCCC3)CCC2)cccc(C(F)(F)F)c1 C(=O)(C(=O)C(C)(C)C)NC(CCOC)C(=O)N(C)CC1(O)CCC1 c1(C(=O)NC(CN(C(C(C)N2CCCC2)=O)C)(C)C)cc(N)cc(O)c1F c1(NC(C2CC2C(=O)NCCC2CC2)=O)cccc(-c2nnnn2C2CC2)c1 C1(N(C(c2ccc(OC)cc2)=O)C)CCN(C(c2c[nH]nc2Cl)=O)CC1C c1(OC)cc(C(=O)NCCOCCN(C(=O)C(C)OC)C)c(C)c(Br)c1 c1(C(=O)NCC2OCC(CNC(=O)CCSc3ccccn3)C2)cnccc1Cl C1(C(N(C(CC(=O)NC2CC(C(C)O)C2)C)C)=O)C2CC3C(C2=O)C13 c1(CCN(C(C(=O)NCCCNCC(=O)NS(CC)(=O)=O)=O)CC)ccccc1 N1(C(CCC#CC)=O)CC2CCN(C(=O)CC(C)P(C)(C)=O)CC2C1 c1(CN2CCN(S(CC)(=O)=O)C(CO)C2)cc2ccoc2cn1 Cc1nc(N(CCNC(=O)Cn2ccsc2=N)C2CC2)ccc1[N+](=O)[O-] C1(C)(CC)C=C(C(=O)N(C2CC(NC(c3cn(C4CCC4)nc3C)=O)C2)C)C1 CCCC(C(=O)NCCC1CC(C)(C)CO1)NC(=O)C#CC1CC1 CC1OC2(C)CC1(C(=O)NCCN1CCN(c3cc(C(N)=O)nc(Cl)n3)CC1)C2 Cc1ccc(OC(C)C(=O)Oc2cnn(C(C)C(=O)OC(C)(C)C)c2)cc1 c1(C(N2CC3(CN(C(c4cc(C)n(C)n4)=O)C3)C2)=O)cn(C(C)C)c(=O)nc1O c1(OC)cc(CC(=O)NCCC2CCN(C(=O)C(C)C(C)(F)F)C2)ccc1Cl C=C(Cl)CC(C(=O)N(C)Cc1nc(C)no1)NC(C1CC2(CC2)CO1)=O CC(C)C1=NOC(C(=O)NCC2CN(C(C3(CO)CCOC3)=O)CC2(C)C)C1 CCC(O)C(F)(F)C(=O)N1CC(O)(CN(C)C(c2ccc(=N)[nH]c2)=O)C1 c1(C2(OC)CCC2)nccc(=NC(=O)c2cc(OC)c(OC)cc2Cl)[nH]1 CC1CN(C(C2(C(N)=O)CC2)=O)CCC1CNC(c1nccs1)=O C(=O)(C(C)(C)CCCF)NC12C(CN(C(C(CCC)NC(C)=O)=O)C1)CC2 Cn1ccc(=O)c(C(=O)NC2CC(CC(=O)NCC3(CC4CCC4)CC3)C2)c1 c1(C(=O)NC2CC3(C(NC(CCC(CC)C)=O)C3)C2)cccc(SC)c1[N+](=O)[O-] N1(C(c2nc(C)n(C)c2)=O)CCOC2(C1)CN(C(C1(C)CC1(F)Cl)=O)C2 CC(C)(C)C#CC(=O)NCc1ncoc1CCNC(C1CC1C1CCCC1)=O c1(CC)c(OC)cccc1C(=O)NC(C)(CNC(=O)C(C)n1cncn1)CC c1(CCC=C)ccc(S(=O)(=O)NCc2cn3ccccc3n2)cc1 N1(C(c2c(C)ccn2C)=O)CCCC(O)(CNC(C2(C)CC2(Cl)Cl)=O)C1 C12(CNC(C3C(C)CCC3)=O)CCCOC1CCN(C(=O)C(=O)c1ccco1)C2 Cc1cc(C(=O)NCC2CC3CCC2N3C(C2(C)CCCCC2)=O)nc(O)n1 CCC(CC(=O)NCC1CC(C#N)C1)N(C(=O)COCCCF)C CCCC(CC(=O)N1CCCC1(CC)CC)NC(C1(C)CCCCC1)=O c1(OCCCCC)cccc(NC(C2(F)CN(C(=O)CN3CCCC3)C2)=O)n1 C1(F)(CNC(c2csc(Br)n2)=O)CCN(C(=O)C(F)CC2CCCC2)C1 CCCCC(O)C(=O)NC1CCN(C(=O)C(C)Oc2ccccn2)CC1O c1(CN2CC(C(N3CC(C(N)=O)OCC3)=O)OCC2)ccc(Cl)c(O)c1 c1(CC)cc(CC(N2CC(NC(C3CC(=O)N(CCOC(C)=O)C3)=O)C2)=O)n(C)n1 CC(C)C1=NOC(C(N2C(C(N3CC(F)(F)CC3CO)=O)CCC2C(C)C)=O)C1 Cc1cc(N2CCC(NC3CCCSC3)CC2)ncc1S(=O)(=O)NC1CCC1 C1(CC(=O)NCCNC(=O)OC)CN(C)CCN1C(=O)CC(C)(O)COC c1(OCC(=O)NCC(CCNC(CCc2cc(C)[nH]n2)=O)O)cc(F)cc(F)c1 Cc1ccc(C(c2nnnn2-c2c(C)cccc2C)NC2CC(OC)C2)c(C)c1 CC1(CNC(c2ccc(Br)o2)=O)CC(NC(C2CN(S(C)(=O)=O)C2)=O)C1 N1(C(CC2(N(C)C)CCC2)=O)CCCC(CO)(NC(C2CCC=CCCC2)=O)C1 C(=O)(C(=O)N=c1ccn(Cc2ccccc2)[nH]1)NCc1c(F)c(N)c(Cl)c(F)c1 N1(C(C2N(C(c3c(CC)c[nH]c3)=O)CCN(C)C2)=O)CCCN(C)CC1C C12(C(=O)NC3CCCCN(C(C(=O)N(C)C)=O)C3)CC1COC21CCC1 N1(C(C2CCCN(C3CC3)C2)=O)CC2(CCN(C(C3(n4cnnn4)CC3)=O)C2)C1 N1(C(C2(N(C(C(C)NC(=O)C3CC3)=O)C)CC2)=O)CCc2sccc2C1 c1(CNC(CNC(CC)=O)=O)ccc(C(C)NC(=O)CCc2ccc(Cl)s2)cc1 C(CC(C(C)C)NC(=O)Cc1ncc(C)s1)NC(C(CC)n1ccnc1)=O CC1CC(NC(=O)CSc2ccccn2)CCN1C(=O)C1=C(Cl)CCC1 C1(O)(C(=O)OC(C)(C)C)CCN(C(=O)C(N)Cc2cccnn2)C1 n1(CC)ccc(C(=O)NCCCOCCC(=O)NCC2(C)CC3CC3C2)c1C CC1(C)CN(C(=O)CN(C(=O)C=CCF)CC2CC2)CCC1O c1(CCC)ncoc1C(=O)NCC1(NC(C2CC=CCO2)=O)CCOC1 C1(O)(CNC(c2ccc(F)s2)=O)CCCN(C(=O)Cc2ccc(Cl)c(F)c2)C1 C(=O)(C(F)(CC)C(=O)OC)NCC1CCCN(C(c2cnc(CCC)s2)=O)C1 c1(C(N2CCC(C(C)OC)CC2)C(=O)NCC=C)scc(C(=O)OC)c1Cl c1(C(=O)NCCOCCNC(C2(n3cccn3)CC2)=O)cc2n(n1)CCO2 CS(=O)(=O)c1cccnc1N1CCC(NC(c2cccn3nccc23)=O)C(F)C1 c12ccccc1C(=O)N2.C1(C)(OCC(=O)N(CCCN(C)C)C2CC2)CCCC1 N1(C(C(CSC)O)=O)CCC2(CCCN(C(=O)C(c3cc(C)oc3C)C)C2)C1 c1(NCCCN2CC(C)CC(C)C2)ncc(S(=O)(=O)N2CCCCC2)cc1Cl Cc1nc(C2CC2)oc1C(=O)NC1CCC(CNC(c2cc(F)c[nH]2)=O)C1 C1(NC(=O)OC(C)(C)C)CCCC(N(C(=O)CCc2cn[nH]c2)CCC#N)CC1 C1(CNC(C(CC)OCC)=O)CC(C(=O)NCC(C)(C)OC)=NO1 c1(C(N2CC(C(C)NC(C=C(COC)C)=O)OCC2)=O)nc(C)c(C)nc1O c1(C(N2CCCC(C)(CNC(C3CCN(CC)C3)=O)C2)=O)cc(F)c(N)cc1F c1(C(N(CCC(C)NC(CCNC(C)=O)=O)C)=O)csc2c(F)cccc12 N1(C(c2c(C)c[nH]n2)=O)CCCCC(CNC(C2CC(N3CCCC3)C2)=O)C1 C(=O)(C1CCCc2nn[nH]c21)NCCCNC(C1C2(CC(C)(C)C2)C1)=O C1(C(C(=O)NCC(C)(C)OCC)NC(=O)OCc2ccccc2)CCC2(CC2)CO1 Cc1ccc(S(=O)(=O)N2CC(O)CC2CN(C(=O)C(c2c[nH]nc2C)=O)C)cc1 S(=O)(=O)(c1cnc(NC(C)Cc2cccs2)c(Cl)c1)N(C(CCSC)C)C [N-]=[N+]=NC1CCN(C(=O)C(C2(O)CCCCC2)NC(=O)C(F)=CC2CC2)C1 c1(C(=O)NC(C2CCN(C(COC)=O)C2)C(=O)O)ccc(S(=O)(=O)NC(C)=O)cc1 C1(C(=O)NC2CN(C(C)C)C(=O)C2)CC12CCN(C(C1CS(=O)C1)=O)C2 C(=O)(CCCCCF)NC1C(NC(c2c(C)n(-c3ccn(C)n3)nn2)=O)CC1 c1(C(=O)NC(C(C)NC(=O)CCS(C)(=O)=O)(C)C)cncc2nnn(C)c12 C(=O)(CCCCCCCC)NC(CNC(CSCC)=O)C1CC1.c1cccc(C)c1 c1(C(=O)NC2CCC(NC(C(COC)O)=O)C2)ccc2ncccc2c1 C1(OC)CN(C)C(C)(C(=O)NCC2CCN(C(c3cc(C)ccc3F)=O)C2)C1 Cc1nnc2cnc(C(N3CC4CC3C4CNC(=O)CCC3CCCC3)=O)cn12 n1(C2CCN(C(=O)NC(c3cc(C)cc(C)c3)C)CC2)c(O)nc2ccccc12 c1(C(N(CCCN(C(C2C(C(C)C)C2)=O)C)C)=O)cc(-c2csc(CO)n2)c[nH]1 C(=O)(C(O)C(F)(F)c1ccccc1)NCC1(C(C)NC(C=CC(C)C)=O)CC1 N1(C(c2cc(CCC)[nH]n2)=O)CCCCC(NC(C23CC(CCO2)C3)=O)C1 C(=O)(C(C)CCCC(C)C)NC1CCN(C(CCOCC=C)=O)CC1CO C1(C(=O)Nc2c(CC)onc2C)CN(C(=O)C(O)C(F)(F)F)CCN1C Cc1c(C(N2CCC(O)(C(C)CNC(C3CC(F)(CF)C3)=O)C2)=O)cccc1N C1(C)(C(=O)NCCC(C)(C)NC(C(C)OCC=C)=O)CC=C(C)CC1 Cc1cccc(CNC(c2cccnc2CNC(=O)C(C)OC(C)=O)=O)n1 N1(C(C=C)=O)CC2(CNC(=O)C(C)C(C)COC)CC1CO2 Cc1nc(C)c(C(N2CCCC2(C)CNC(c2c(C)noc2C)=O)=O)s1 C1(C(=O)NC2C(C)N(C(c3cccc(C(F)F)c3F)=O)CC2)CC12CCSCC2 CN(C)NC(=O)CCC(=O)N1CCC2C(C(N3CC(O)CC(O)C3)=O)C2C1 Fc1cc(F)c2cccc(-c3nc(C(c4ccc(C(F)(F)F)cc4)F)no3)c2n1 C1(NC(c2cccc3c2OCO3)=O)CC2CCC1N(C(C1CCCNS1(=O)=O)=O)C2 CC1=C(C(=O)NC2CCC(CNC(c3oncc3C)=O)CC2)SCCO1 C(=O)(C(C)C(=O)N1CCC(CCNC(C2CC(C)(C)CO2)=O)CC1)OC c1(C(C)=O)cn(C)nc1C(=O)NCC(C1CC1)NC(c1cc(C(C)C)no1)=O C1(C(=O)NCC2C(C)CN(C(=O)CC3CC3)C2)OCC2COCCC12 c1(CC)c(C(=O)NCCC2(O)CN(C(=O)CC(C3CC3)C3CC3)C2)nnn1C CCC(C)C(=O)NCCC1CCCN1C(C1CC(F)(CF)C1)=O C#Cc1ccc(C(N2CCN(C(C3CCC4CC4CC3)=O)CC2)=O)cc1C N(C(=NCC(C)N(C)C1CC1)N1CCC2(CC1)CCS(=O)(=O)CC2)C(CC)C CC(C)C(C(=O)NCC1CSCCS1)NC(c1cccs1)=O C1(c2ccccc2)(CNC(C2C(C)CC2)=O)CC(NC(c2cnc[nH]2)=O)C1 N1(C(CC(C)O)=O)CCc2nc(C(N3CCC(C#N)(CO)C3)=O)cn2CC1 C(=O)(CCC(C)(C)[N+](=O)[O-])NCC(CNC(C(C)C1CCOC1)=O)S(C)(=O)=O CCC(CC(=O)NCCCCCNC(=O)Cc1ncn(C)c1C)SC Cc1cc(O)c(C(=O)N(C)CC2CCCN(C(=O)C(C3CC3)C3CC3)C2)nn1 c1(C(=O)NCC2N(C(CNC(C)=O)=O)CCCC2C)cc(O)ccc1[N+](=O)[O-] CCCCC(CNC(=O)CC(C)(C)c1cccs1)N1CCOCC1 N1(C(CSCCCC)=O)CC(NC(c2cc(C)n(C(C)C)c2)=O)C(N=[N+]=[N-])C1 CCS(=O)(=O)CC(=O)N1CCCC1C1CCN(C(=O)CN2CCS(=O)CC2)CC1 c1(-c2cn(C3CC(C(N(C4CCC4)CC)=O)C3)nn2)ccc(F)cc1 CCCCC(O)CCC(=O)N1CCC1CNC(C1(O)CCCCC1)=O c1(C(N2C(C(C)C)C(NC(C3CC(O)C3)=O)CC2)=O)ccc2sccc2c1 C1(NC(C2(C(=O)NC)CCC2)=O)CCN(C(c2ccsc2Cl)=O)CC1C c1(C(=O)NCC(CNC(C2C(OCC)C2)=O)F)cc(OC)c(OC)c(Cl)c1 N1CCCCC(O)C1=O.C1(F)(CNC(C2CCCN2C(=O)C2CC2)=O)CN(C=O)C1 NS(=O)(=O)C1CC(C(N2CCN(C(c3ccc(O)cc3)=O)C(C3CC3)C2)=O)C1 C#Cc1cccc(C(=O)NC(C)(CNC(=O)C(C)=CC=C)C2CC2)c1 c1(C(N2CCC(NC(C3N(CC)C(=O)CC3)=O)C2C)=O)ccc(=O)n(O)c1 Cc1cnn(CC(=O)NC2CCCN(C(=O)CC3C=CCC3)CC2)c(=O)c1 c1(N(C)CC)nc(=NCC(CO)C2CC2)[nH]c2cc[nH]c12.N12CCC(C1)C2 c1(CCC(=O)NCC(C)(C)NC(CC(C(CC)C)O)=O)ccc2cnn(C)c2c1 CC(C)CCC(F)C(=O)NCC1(O)CCCN(C(C23CCN(CC2)CC3)=O)C1 N1(C(=O)OC)CCCC(C(=O)NC2CC(CCNC(C3CCOCC3)=O)C2)C1 c1(NC(C2CC(F)CN2C(=O)CSc2ccncc2)=O)c(Br)cccc1[N+](=O)[O-] N1(Cc2cnc(SC)nc2)CCN(C(c2ccc(I)cc2O)=O)C2CC12 N1(C(C(C2CC2)SC)=O)CCN(C(=O)C(N2CCCC2)C2CC2)CC1C c1(OCC#C)ccc(C(N2CC(CNC(c3sccc3C(F)F)=O)C2)=O)cc1 C1(CNC(=O)C=Cc2ccncc2)CCCCN1C(=O)CCCc1ccncc1 N1(C(CC=CC=C)=O)CC(C(N2CCCC(C#N)C2)=O)C2(CCC2)C1 C1(C)(CC(=O)NC(c2ccccc2)C(=O)NCc2cc(CC)on2)CCOCC1 Cc1cc(SCC(N2CCCC2c2ccncc2)=O)cc(C)c1 C1(NC(C2(CN(C)C)CC2)=O)CCCC1CNC(=O)C(C)(C)C1CC1 CC(C)C(O)C(C)(C)C(=O)NC1CCCC1NC(c1cc(O)cc(O)n1)=O O=C1CC(C(=O)NC2COCC2NC(c2ccnc(N3CCCCC3)c2)=O)=NN1 c1(NC(C(=O)NCC(c2ccccc2)NC(=O)CCF)=O)ccc(F)cc1F CCCC(O)CC(=O)NCC12CC(NC(=O)CSCC(N)=O)(C1)C(C)O2 c1(CC(=O)NC)csc(CCNC(=O)NCCOC)n1 CC(C)C(C(=O)NCCC(C(C)C)NC(c1c[nH]nc1C(N)=O)=O)n1cnnc1 C1(NC(C(C)CC2CCCC2)=O)CCN(C(c2cnc(N(C)C)nc2)=O)C12CC2 c1(C(=O)NC(C2CCN(C(CC3N(C)CC=CC3)=O)C2)(C)C)ccc(N)c(N)c1 CC1(C)C(NC(C2CC(=O)N2)=O)CCN1C(c1cccc(N(C)C)n1)=O S(=O)(=O)(c1ccc(F)c(F)c1)N1CC2C(NC(c3cc4n(n3)CCC4)=O)C2C1 c1(N2C3(CNC(c4ccnc(C)c4C)=O)CC(C2)C3)ccc(S(C)(=O)=O)cn1 CC(CCC(C)(C)C)C(=O)N1CCCC(N(C)C(c2ccnn2C2CC2)=O)C1 N1(C(CCC2CC(NC(C3N(C)CCCC3)=O)C2)=O)CC2(CCNC(=O)O2)C1 C=CCCCC(C(=O)NC1CN(C)CC12CC2)NC(c1cocn1)=O c1(CNC(c2ccc(Cl)cc2)=O)cc(O)nc(CNC(C23COC(CF)(C2)C3)=O)n1 C(=O)(C(O)CC(F)(F)F)NC1(CC=C)CN(C(c2ccc(O)c(Cl)n2)=O)C1 C1(N)(C)CCCCCC1.C(=O)(C(C)n1cccn1)C(N(CC)CC1CC1)=O c1(C(N(CC(=O)Nc2ccc(CC)nc2)C2CC2)=O)cccc2ccnn12 C1(CNC(C2(CC(C)C)CCC2)=O)CC(O)CN1C(c1cnc(Br)s1)=O c1(C(=O)OC(C)C(c2ccccn2)C)cc(OCc2cnn(C)c2)cc(Br)c1 N1(CCC#C)CCN(C(C2(C)CC(NC(=O)C(C)N3CCCC3)C2)=O)CC1 N1(C(CN2CC(C)C2)=O)CCC2C(CCN2C(=O)C#CC2(C)COC2)C1 C(=O)(CC1=CCOCC1)N1C(CN(C(=O)C=Cc2ccsc2)C)CC(F)C1 C1(C(C)C)C(C(=O)N(C)CC2CC(F)C2)CCN1C(=O)CC1CCC(C)(C)C1 c1(-c2n(C3C(C)OCC3)nc(-c3cccnc3)n2)cc2n(c1)CCS(=O)(=O)C2 C1(CCNC(CCCC(N)=O)=O)CCN(C(=O)CC2CC3(CC3)C2)CC1(F)F c1(C(=O)NCC2(C)CC(NC(=O)CCSC(F)(F)F)C2)cnc2ccccn12 c1(C(=O)OC)sc(C(N2CCC(O)(CNC(c3c(C)ccn3C)=O)C2)=O)cc1C C(=O)(CCCCc1ccccc1)NCC1(OC)CCN(C(=O)COC(C)(C)C)C1 c1(C(=O)NC2C(CNC(c3c(C)c[nH]n3)=O)C2)cc2ccc(Br)cn2n1 C(=O)(C1=CCCC1)NCC(C(C)C)NC(c1cnoc1-c1cccs1)=O C1(C(=O)NC2(C)CN(C(c3ncn(CC)n3)=O)C2)CN(CP(C)(C)=O)C1 C1(NC(c2c(C#C)cn(C)n2)=O)CN(C(c2sccc2OC)=O)CC1C1CC1 Cc1cc(C(=O)NC(CNC(=O)C(F)(F)c2csc(C)c2)C2CC2)co1 N12CCC3(CC3C1=O)C2.c1(NC(C2CCCCC2)=O)cc(OC(F)F)ccn1 N1(C(C2CC(OC)C2)=O)CC(O)C(O)C1CNC(c1cc(C)[nH]n1)=O C1(NC(C(CC=C)C)=O)CC(F)CN(C(c2ccccc2Br)=O)C1 c1(CC)ccc(C(=O)NCc2csc(CNC(C3CC3c3ccccc3)=O)n2)[nH]1 C=CC(C)C(=O)NC(C)(CNC(=O)C(C)(C)C1CCCC1)Cn1cccn1 c1(CC(C)C(N2CC3C(NC(c4cn(C)nn4)=O)C3C2)=O)cccc(Br)c1 c1(C(=O)NC2C(NC(C(F)=CCC)=O)CC2)cnnc(C)c1 c1(C(=O)NCC2CC(NC(C3(CCF)CC3)=O)C(O)C2)c(F)cc(F)cc1Cl N1(C(c2nc(CC)sc2)=O)CC(NC(=O)C(C)CC(N)=O)C2CCCC12 CC1C(NC(c2cccnn2)=O)CCN1C(C1CC2CCCC12)=O c1(C(N(C2CS(=O)(=O)C2)C)=O)ccccc1SC(F)F C(C(=O)NC1CCC1C(=O)NC(C)(CO)C1CCCC1)(C(C)(C)C)OC CCC(CC(F)(F)F)NC(c1cn(CCNC(c2ccc([N+](=O)[O-])o2)=O)nn1)=O CCC(CC(=O)N1CC(CNC(C2CC2(F)F)=O)(OC)C1)C1CC1 C(=O)(C1=CCC(C)(C)CC1)NCC(CN(C)C(c1cc(F)n(C)n1)=O)(C)C N1(C(C(COC)C)=O)CC2CC2(NC(c2ccc(-c3nccs3)cc2)=O)C1 C1(CNC(C(OC)OC)=O)CCCCN1C(=O)CC1CCCOCC1 C=CCC(C)(C)CCNC(C1(NC(C2CC(=O)C2(C)C)=O)CCSC1)=O C#CCN=S(C)(=O)NCCCC(F)(F)Br.c1ccccc1 C1(NC(=O)CC2CCS(=O)(=O)C2)CCOCC1NC(=O)CCOCC1CC1 C1(C(N2CC(CCCCNC(=O)C(C3CC3)C3CC3)C2)=O)CCCCS1(=O)=O c1(CCC)c(C(=O)NCC(c2ccccc2)Nc2nccc(SC)n2)cnn1C Cc1cc(Cl)cnc1NC(N1CC(CC(=O)N(C)C)C1)=O c1(C(=O)NCC2(C(=O)NC3CC4(CCC4)C3O)CCC2)cccc2cncn12 C(=O)(CCCCC(N)=O)N1CCC(CN(C)C(c2nn(C)c(=O)n(C)c2=O)=O)C1 C1(Nc2c(OC)cncn2)CCC2CN(C(=O)COCC3CCOC3)CC12 C1(S(C)(=O)=O)(C(N(C)CC2CN(C(=O)CNC(=O)NC3CC3)C2)=O)CC1 C1(CN(C(=O)CCCn2cc(C3CC3C3CCOCC3)nn2)C)CC(O)CN1C C1(O)(C(=O)NCCCC(C)NC(c2cc(=N)[nH]c(=N)[nH]2)=O)CCCCCC1 c1(C(N2CC3(C(NC(C(C)O)=O)CCC3)C2)=O)ncnc2c1cnn2C C1(NC(CC(CC)CC)=O)CCC2(CC1)CC(NC(=O)C(CO)OC)C2 CC1CC(O)CCN(C(C23COCC2CN(C(=O)OC(C)(C)C)C3)=O)C1 CC(CC(=O)N1CSCC1C(N1CCCC(C)C1CO)=O)CC(C)(C)C C1(NC(CC(CC)C)=O)CC2(CCCN(c3ncc(Br)c(C)n3)C2)C1 c1(C(=O)NCC(C)N(C(=O)COC2(C)CCCC2)C)cc(Cl)nnc1O CC(C)CCCOCC(N1CCC1(C)CC(=O)NCC1CC(CN=[N+]=[N-])C1)=O CCCC(CC1CCCC1)C(=O)N1CCCN(C(c2c(C)nn(C)c2OC)=O)CC1 c1(CN(C(C(=O)NC(C2CCCO2)C)=O)Cc2cccc(O)c2)ccc(F)cc1 N(C1COc2c(F)cccc21)C(C(=O)N(C)CC1CCN(c2ccccc2)C1)=O c1(CC(=O)NCC(CO)NC(C2Cc3ccccc3O2)=O)ccc2[nH]ccc2c1 N1(C(C(C)SCC)=O)CCN(C(c2cc(O)cc(O)n2)=O)CC12CCC2 C1(C(=O)NCCCC2(NC(c3nc(COC)sc3)=O)CC2)CC(C)(C)OC1(C)C C1(F)(CNC(=O)NC2CCCC2c2ccc(Br)cc2)CCOCC1 c1(C(=O)NCCN(C(c2c(C)cnn2C)=O)C2CC2)cc2cccnc2cc1F N1(C(c2n(CC#C)ccc2)=O)CCC2CC1CN(C(=O)CNC(N)=O)C2 c1(C(N2CCN(C(c3cc(C)nn3C)=O)CC2CF)=O)cc2c(O)cccc2[nH]1 C#CCC(O)C(=O)N1CCC(CN(C(=O)COCC(=O)OC)C)C1 c1(C(N2CCCC(CCC(N3CCOC4CC34)=O)C2)=O)c[nH]ccc1=O c1(C(=O)NCC2(CCNC(C3C(C)(Br)C3)=O)CC2)ccc(OCF)cc1 C1(NC(CCC(=C)C)=O)CCN(C(c2nc(CC)ncc2Cl)=O)CC1F c1(NC(CC)CCCO)ccc(S(=O)(=O)NCCN2CC3CC3C2)cn1 C1(C)(CNC(C(CC2CC2)OC)=O)CC(F)(F)CN1C(=O)CCSC c1(C(N2CC(NC(C(C)n3cnnn3)=O)(CO)C2)=O)oc2ccccc2c1CO N1(Cc2c(C)c(F)c(F)cc2)CC2OCCN(C(c3ccccc3Cl)=O)C2C1 Cc1cn2c(n1)CCC(NC(=O)Nc1cccc(-c3ccc(C)c(F)c3C)n1)C2 N1(C(CCc2c(C)noc2C)=O)CCN(C(C2CC3C=CC2O3)=O)CC1CO CCCC(C)CCN=c1[nH]c2c(c(=NCC(C3CCCCC3)N(C)C)[nH]1)CSC2 C(=O)(CS(=O)(=O)C1CCCC1)N1CCC(C2CC2)(CNC(CCC(C)C)=O)C1 C1(CC)COC(C)(C)CN1C(C1CCN(C(=O)C(CN(C)C)CC)CCO1)=O C1(NC(C(C)CC2CC2)=O)CC2CC1N(C(c1ccnc(OC(F)F)c1)=O)C2 Cc1c(Br)ccnc1N1CCN(C(=O)C(N2CCCC(O)C2C)=O)CC1 C1(C(N2CCC(CCNC(=O)CCc3cc(C)[nH]n3)C2)=O)(COC)CCCC1 N1(C(C(C)CC2CC2)=O)CCC2(CCC(NC(=O)CN3CCCCCC3)CC2)C1 c1(C(=O)NC(CC(C)NC(CCCC)=O)C)c(OCCOC)cccc1Cl c1(CNC(C(C)NC=O)=O)cc(C(=O)NC(c2ccccn2)C)cs1 Cc1cc(CC(=O)NC2(CCNC(=O)CC3CC4CC4C3)CCCC2)ccc1O C(CCS(=O)(=O)c1ccccc1)NC(C1(N)CC(F)(F)C1)=O C(=O)(C1=CC2CCC1C2)N1CCN(C(c2scc(C#N)c2)=O)CC1CC(F)F c1(C(=O)OC)cccc(-c2ccc(NCc3ccc(C(=O)O)s3)cc2)n1 N1(C(C(COC)C)=O)CCC2C1CCCN2C(=O)COCP(C)(C)=O c1(NC(C)CCNC(c2ccc(Cl)nc2Cl)=O)nc2c(cc1C#N)CCC2 C12(NC(=O)CC3CCOCC3)CCN(C(c3ccc(O)nn3)=O)CCC1C2 C(CC(=O)NC1COC(C(C)C)C1)(C(F)(F)F)NC(c1c(OC)scc1)=O c1(-c2nc(NC(=O)NCc3ccnn3C3CC3(F)F)sc2)c(F)cccc1F N1(C(C(c2ccccc2F)(C)C)=O)CC2(CCC2NC(C2C=CCC2)=O)C1 c1(C(=O)NCC2N(C(CCCOCCOCC)=O)CC2)ccc(Cl)c(S(C)(=O)=O)c1 C1(C#N)(C(=O)NC(CNC(c2c(C)scn2)=O)C(C)(C)C)CC2CC2C1 N1(C(c2c(C)onc2)=O)CCN(C(=O)CCCC(F)(F)F)CC12CCC2 C1(CNC(CC2C(C)C2(F)F)=O)CN(C(c2cnn(CC3CC3)c2)=O)CCCO1 c1(CC(=O)N(CCC(C)NC(Cn2c(C)ccn2)=O)C)cnccc1C(F)(F)F N1(C(Cc2ccc(C)o2)=O)CCOCC(CNC(c2cc(C(F)(F)F)cs2)=O)C1 CC1CC(C(N2CCC(CCN(C(=O)C=CI)C)CC2)=O)CCO1 CCCCC(F)C(=O)NCC1CCC(NC(C2CCCN(C)C2)=O)CC1 C(=O)(NN1CCCC(C(=O)O)C1)C1(N)CCCN(C(C)=O)C1 N1(C(CC(CC)O)=O)CCCCC2(CCN(C(=O)CC3CCC4(CCC4)O3)C2)C1 N1(C(CC(CC)OC)=O)CCCC(C2CCN(C(=O)CCc3cnc(C)o3)C2)C1 c1(C(=O)NCCN(C(=O)C(C)Cc2cnc[nH]2)CC)cc(C)cc(Br)c1 c1(C(=O)NC(C(C)NC(CCOCCOCC)=O)C)cnc(C)s1 c1(CC(=O)NC(C2(NC(=O)Cc3cccs3)CCC2)C)noc2ccccc12 C(=O)(C(C)CC(=O)NCC1CCCN1C(=O)COCc1ccnn1C)OC N1(C(C(C)C#N)=O)CC2(CCC(CNC(=O)C=CC3CCCC3)O2)C1 N1(C(CC(CC)C)=O)CC2(CNC(c3cn(CCCF)nn3)=O)CC1CO2 N1(c2ncc(C(=O)OCC)cn2)CC2CCCN(C(=O)C(F)CC)C2C1 c1(C(=O)NC(C)CCN(C(=O)Cc2ccn(C)n2)C)ccccc1C1CCC1 Cc1nn(C)cc1C(=O)NCC(C)(F)CNC(=O)C(C)NC(N)=O C(CC(=O)NCCN(C(c1cnn(C(F)F)c1)=O)CC)(C1=CCCC1)OCC C(=O)(C(C)(C)C1=CCSCC1)NCCC1CCC(NC(CC2(C)CC2)=O)C1 N1(C(CN(C(C(C)C)=O)C)=O)CC(C(=O)NCCN2CCCCC2=O)CC(C)C1 Cc1ccc(I)cc1NC(C1CCCN(C(=O)Cc2cccs2)C1)=O C=CC1CN(C(=O)C(C)SCC)CC1NC(c1ccc(F)s1)=O CC(CNC(c1ccc(Cl)o1)=O)CC(=O)NC1CC12CC(O)C2 C1(CNC(C(C=C)O)=O)C2CCCC1N(C(C1CCC(C)O1)=O)C2 Cn1ccnc(Nc2cccc(NC(c3cnn(CCN)n3)=O)c2)c1=O C1(NC(c2nc(CCC)oc2)=O)CC2CCC1N2C(=O)CC(C)c1ccco1 N1(C(c2c(NC)cccc2)=O)CCC2C1CCCN2C(c1nn(C)c(C)c1Cl)=O c1(NC(=O)NC(C(CC)C)CO)ccc2nc3n(c(=O)c2c1)CCCC3 C(=O)(CN=c1cc[nH]cc1)N1CCC(CC=C)(C(N(C)CP(C)(C)=O)=O)C1 C1(O)(CNC(C(C)NC(c2c(C)occ2)=O)=O)CCCN(Cc2ccccc2)C1 CC1Cc2sc(C(N3CC(NC(c4cccc(O)c4Cl)=O)C3)=O)cc2C(C)C1 N1(C(c2cc(OC)nn2C)=O)CCN(C(C2CCC(=O)N2C)=O)CC1CC(F)F CC(C)(C(=O)NCCCC1CCOCC1)NC(=O)CC1COCCO1 C1(NC(CCC(=C)Br)=O)CCC2(CC1)CN(C(C1CCC1)=O)CCO2 c1(C(N(C(C)CCNC(c2c[nH][nH]c2=N)=O)C)=O)ccc2c(O)n[nH]c2c1 c1(CC)ccc(C)c(C(=O)NC2(CCCNC(=O)C(O)C(C)C)CC2)c1 Cc1cc(C)c2cc(C(N3CCC3CNC(=O)C3=CCCOCC3)=O)[nH]c2c1 CCCC(C#N)C(=O)N1CC2(CC(NC(=O)C(C)OCCC(C)C)C2)C1 C(=O)(CN=S(C)(C)=O)NC1C(NC(C(c2ccc(OC)cc2)CC)=O)CCCC1 C1(CNC(C=CC=CC)=O)CCCC(CNC(c2cc(CC)ncn2)=O)C1 Cn1cc(CCC(=O)NCC(O)CNC(C2(CO)CCCC2)=O)nn1 C(=O)(C1=NOC2(CCOC2)C1)N1C(CNC(c2ccn(CCF)n2)=O)COCC1 CCC(O)C(C)C(=O)NCC1(NC(c2cn(C)nc2Cl)=O)CCCC1 N(C1C(=O)Nc2c(Br)cccc21)C(N1CCc2cc(Cl)nnc2C1)=O C(N=c1[nH]c(=NCc2cccs2)c2ccccc2[nH]1)C1C(CCC)CCC1 C1(O)(CCNC(c2csnn2)=O)CCN(C(c2ccc(O)c(F)c2)=O)CC1 c1(C(=O)NC(C=C)CO)cn2c(C)ccc(-c3cccc4c3OC(F)(F)O4)c2n1 c1(OCC)cc(C(=O)NCC2CN(C(c3csc4cncn34)=O)C2)ccc1OC c1(N(CCCCCCC)CC)nc(=NC(C)c2nncs2)[nH]c2c1CCC2 c1(CC)nc(C)oc1C(=O)N(C1CN(C(=O)C(CC2CC2)OC)CC1O)C C1(C(=O)NCC(CNC(=O)CCCSC)OC)(OC)CCC12CCC2 N1(C(C=C(C)C2CC2)=O)CC2(CCC(NC(=O)Cn3cc(C(C)O)nn3)CC2)C1 c1(N(C)C)ccc(C(=O)NCCOC2CCN(C(=O)C(C)(O)C3CC3)CC2)cc1 c1(CN2CCC(NC(C3CCN(CC)C3)=O)C(O)C2)cc2c(OC)cccc2[nH]1 Cc1csc(C=CC(=O)NCC2CC(CNC(=O)CO)CO2)n1 C1(CNC(C(F)OC)=O)CCN(C(c2ccc(C)nc2O)=O)C12CC2 N1(C(C2CN(C)C2)=O)CC2(CO)CC1(C(N1CCC=C(F)C1)=O)C2 c1(C(N(CCNC(C2N(C=O)CCC2)=O)CC2CC2)=O)cc2sccc2[nH]1 C#Cc1cc(C(N2CCC(CNC(C3(c4ccn(C)n4)CC3)=O)C2)=O)cc(Cl)c1 N(C1CCCc2ccc(F)cc21)C(N1CCC2(CCCNC2)C1)=O C1(c2n(C)cnc2)CN(C(=O)CNC=O)CC1CNC(c1cnc(C(F)F)s1)=O N1(C(CC(CCC)O)=O)CCC2(CCC2)C(NC(c2cnc(OCC)cn2)=O)C1 C1(C(C)C)CN(C(C2(F)CCN(C(=O)CC3(C)CCOCC3)CC2)=O)CCCO1 c1(OC)ncc(NC(C2(C)CCCN2C(=O)CN2CCOC2=O)=O)cc1Br c1(OCC(=O)NCCCCN(C)C(C2CCC3CC23)=O)cccc(F)c1F C1(C(N(C(CCNC(C2ON=C(CC)C2)=O)C)C)=O)CC2CCC1CC2 c1(OCCCC)ccc(C2(C(=O)NC3CC(NC(=O)C(F)(F)C4CC4)C3)CC2)cc1 C(=O)(C(C)CC(N)=O)NCC(N1CCN(C(CC=CCC)=O)CC1)=O c1(CCNC(C2CC2Cl)=O)c[nH]c2ccc([N+](=O)[O-])cc12 c1(C(N2CC(C)C(NCc3ccc(O)cn3)C2)=O)cccc(O)c1[N+](=O)[O-] N(C(=NCCOC1CC1)N1CCS(=O)(=O)C(C)(C)C1)CC(C)(C)C N1(C(c2ccc(CC)nc2)=O)CCC(O)C(C(=O)Nc2ncc(O)cc2Cl)C1 c1(C(N2CC(OC)(CNC(c3scnc3C(C)C)=O)C2)=O)cc(F)cc(C)c1N N1(C(C(C)N2CCC2)=O)CCOCC(F)(CNC(=O)CCc2cn[nH]c2)C1 c1(OC)ccc2[nH]c(=NCCc3c[nH]nc3C)nc(N3CCSC(C)(C)C3)c2c1 CCC(CC(=O)N1CCCC(CC)(NC(=O)CCSc2ccccc2)C1)C(F)F Cc1cnc(CN2C(C(N3CC4CC4C3)=O)CC3CC23)c(F)c1 c1(C(N2CCC(C3N(C(C(F)OC)=O)CCC3)C2)=O)nc(Cl)sc1Cl c1(C(N2C3C(NC(CCC(=C)C)=O)C(CC3)C2)=O)c(C2CC2)nc2sccn12 Cc1ccc(Cn2cc(CN(O)C(=O)C3CNC(=O)N3)nn2)o1 C(=O)(C(C)(C)C(C)(F)F)NC(C1CC(NC(c2c(C)occ2)=O)C1)C C1(NC(c2c(C)[nH]nc2C(C)C)=O)CCN(C(=O)C(=O)N(C)C)C(C2CC2)C1 C1(C(=O)NC(C)CCNC(=O)CC2CC2(Cl)Cl)CCOC2(CCCCC2)C1 C1(OC)(OC)C(C(N2CCC(C(=O)OC)CC2(C)OC)=O)CC1(F)F Cc1ncc2c(n1)CN(C(c1cccc3nc(C(F)F)sc13)=O)CC2 CCCC(CC)C(c1nnnn1CC(F)F)NCc1cnccc1C CC(C)(COC1CCCC1)C(=O)NC1CCOCC1NC(c1cnsn1)=O CC1(C)CC(CNC(=O)C(CCF)NC(C2CC3(CCC3)C2)=O)CCO1 C(=O)(CCCCC(F)F)NCC1CC(O)(CNC(=O)Cc2nnc(O)s2)C1 c1(C(N2CC(O)CC(NC(CCC(C)N(C)C)=O)C2)=O)ccc(F)c(Cl)c1F c1(C(=O)NCC(CC)NC(C2CC3CCC2O3)=O)ccc([N+](=O)[O-])cc1 c1(C(=O)NC(CNC(c2nc(C)sc2)=O)(C)CO)cccc2occc12 C(=O)(CN=c1cc[nH]cc1)N1C(C(=O)N(c2ccccc2Cl)CCO)CC(O)C1 C(CCC(=O)N=c1ccn(C2CCC2)[nH]1)NC(=O)CC=Cc1ccccc1 CC(C(F)C(=O)NC(C)CC1CN(C(c2sccc2C2CC2)=O)C1)C(F)(F)F c1(C(=O)NCC(C(C)(C)C)NC(c2cn(C)c(=O)cc2)=O)cccn2cncc12 C1(C(N2C(C)(CCC)CC2)=O)CC(C)CCN1C(c1cc(O)nn1C)=O C1(CNC(C(=O)N(CCC)Cc2ccc(Br)cc2F)=O)CC12CCOCC2 c1(C(=O)OC)cc(C)c(C(=O)NCCCN(C(=O)Cc2cnn(C)c2C)C)o1 c1(C(N2C(CNC(c3cc(C(C)(C)C)n[nH]3)=O)CCC2)=O)cccc(=O)[nH]1 c1(OCC)cccn2ncc(CS(=O)(=O)NC(c3nc(C(C)(C)C)no3)(C)C)c12 CC(=O)CCCC(=O)NC(C(=O)NCc1cc(=O)cc[nH]1)C(C)C c1(C(N(C(CC)CNC(=O)CC2CNC(=O)C2)C)=O)ccc(C)c(C)c1F N1(C(c2c(C)nc(CO)o2)=O)CCCCCC1CNC(c1ccc(C2CC2)o1)=O c1(NC(=O)CC2C(NC(c3ccsn3)=O)CC2O)cnn(C(F)F)c1C1CC1 CC(CS(=O)(=O)Nc1ccc(N2CC(C)(O)C2)cc1)C(C)(F)F c1(CNC2CC(NC(c3c(C)ncs3)=O)C2)cc([N+](=O)[O-])c(Cl)cc1F N#Cc1c(Cl)nc[nH]c1=NCC(CNC(=O)C=Cc1ccccn1)C(F)(F)F N1(C(C(=Cc2cn[nH]c2)C)=O)CC(CNC(C2CC2(F)Cl)=O)CC1(C)C N1(C(c2c(C)nn(C)c2)=O)CCCC(O)(CCNC(C2C(C)C2C)=O)C1 c1(C(=O)NCC2CCCCN(C(CCC(C)(C)F)=O)C2)cc2n(n1)CC(F)C2 c1(NC(c2cc(C)[nH]c2)=O)c(-c2ccc(F)nc2F)ccc2c1OCO2 C1(NC(c2n(C)ccn2)=O)CN(C(=O)C(C)(C)C(N)=O)CC12CCC2 C(=O)(C1=NOC(C2(O)COC2)C1)N1C(C)(CN(C(C2CNC(=O)N2)=O)CC)CCC1 C=CC(C)CCNC(=O)CCCC1(NC(=O)CCc2cscn2)CCC1 CCC(CC(F)(F)F)OC(c1cnn(C2CC2(F)F)c1)=O c1(CN2CCC(F)(CNC(C(C(=O)OC)C)=O)CC2)cc(F)c(C)c(Br)c1 CC1(C)CCCC(C(N2CCC(C(F)F)C2)=O)C1 N1(C(c2sccc2F)=O)CCN(C2CN(C(c3[nH]nnc3C3CC3)=O)C2)CC1 C1(C(=O)NCC(CC)NC(=O)C=C2CCC(C)C2)(OCC)CCCCCC1 CC(C)(CCCNC(C1CC(C)(C)C1)=O)NC(C1CC1C(F)(F)F)=O c1(NC(N)=O)ccc(Cl)c(C(N2CC(NC(C3CCCCNC3=O)=O)C2)=O)c1 C1(C(=O)NC2C(NC(c3ccc(-c4ccccn4)s3)=O)CC2)CCC=CCCC1 C(c1cnn(C)c1)=CC(=O)N(CCC(=O)NCC(O)C1CC1)C C12(CNC(CC3(C)CCCO3)=O)CCC(CC1)N(C(c1ccnn1C(F)F)=O)C2 Cc1ccc(OCC(=O)NC(CNC(c2ccc(=O)n(C)c2)=O)C2CC2)c(Cl)c1 N1(C(C(F)OC)=O)CC(CNC(C2(CCF)CCOCC2)=O)C2(CCOCC2)C1 N1(C(C)=O)CCCCC1CNc1c(C)cnn1C1CCN(Cc2nccs2)CC1 n1(CC(=O)NC(CC)(CNC(=O)Cc2cnc(C3CC3)[nH]2)CC)nc(C)ccc1=O C1(C)(C(=O)NC(CC)(CNC(=O)C(F)CN(CC)CC)CC)CC2CCC1C2.CC N1(C(CCCCCCC)=O)CC2COCC(C1)C2NC(c1coc(CC)n1)=O C(=O)(N=c1ccn(CCCO)[nH]1)C1(CC)CCN(C(=O)C=CCOC)C1 CCCC(CCC)=CC(=O)NCC1CC(C(N2CC(F)(CC)C2)=O)C1 c1(C(=O)NC(CC)CC2CC2)ccc(C(F)(F)F)nc1C(F)(F)F N1(Cc2c(C(=O)OC)n(C)nn2)CCC(N2CCN(C)CC2)CC1C C=CC(C)(C)CCCNC(=O)C(F)C1CC(NC(c2cc(C)c(C)s2)=O)C1 N1(C(CCN(C)C(c2csc(O)n2)=O)=O)CCC(CF)CC1 C(=O)(C1=CCCN(Cc2cc(F)cc(Br)c2F)C1)NC(CC=C)CO CC1(NC(c2ccc(C(F)F)cn2)=O)CCN(C(=O)C=CC(N)=O)C1 C(=O)(C(C#N)C(C)(C)C)N1C(C)(C(=O)Nc2cccc(C)c2F)CCC1 c1(CC)cnc(Cl)[nH]c1=NC1CCCN(C(=O)Cn2nc(C)cc2C)CC1 C(=O)(C(C)(CO)NC(=O)Cc1ccoc1)N(C(CC)CC)C C1(NC(c2nc(OCC)oc2)=O)CC12CCC(NC(c1oc(C)nc1C)=O)CC2 c1(CC)ncccc1C(=O)NC(Cc1cnc[nH]1)C(=O)N(CC(C)CO)C c1(NC(C2CCN(C(c3c(C)oc(Cl)n3)=O)C2C)=O)ccc(O)c(Cl)c1 CC1CN(C(C2(C)CN(C(=O)CC3CCCN(C)C3)C2)=O)CCCO1 Cn1ncnc1CCCNC(=O)C=CCC1(N(C(=O)CSC(F)F)CCO)CCC1 C(CC(=O)NNC(=O)c1cc2ccccc2[nH]1)(C(F)(F)F)OC(C)(C)C O=C(C(O)CCCNC(=O)Cc1ccccc1F)NCc1cccc(F)n1 c1(CCNC(=O)C=CCNC(=O)CC2(O)CCC2)ccncn1 c1(C(N2CCCC(C(=O)NC3CCS(=O)(=O)C3)CC2)=O)c(O)cc(O)cc1O c1(C(N(C2CCN(CC3CCCO3)CC2)CCN(C)C)=O)ccc(O)c(CO)c1 c1(C(=O)NCC2N(C(c3c(OC)nccc3)=O)CC(OC)C2)ccnc(O)c1F C1(C(N2CC(O)(C(C(=O)NCc3scc(C)n3)F)C2)=O)CCC(=O)NC1 Cc1c(C(c2c(Cl)cccc2Cl)=O)cc(CCC(=O)N(C)C)n1C c1(C(=O)NC2C=CCN(C(C3(CC)CCC(O)CC3)=O)C2)ccn2ncnc2c1 c1(C(=O)NC(C(CO)NC(c2c(OC)noc2C)=O)C)ccccc1S(C)=O C12(C(=O)NC3CCN(C(CC4(CC=C)CCCC4)=O)CC3)CCC(F)(CC1)CC2 c1(C(=O)NC2CCCN(C(C3CN(C)C(=O)N3)=O)C2)ccc2oc(S)nc2c1 C=Cc1ccc(C(=O)NC2CC3(C2)CC(Nc2ncncc2I)C3)cc1 CCCCC(CC(=O)N1CCCCC1CF)NC(C1C(C)C1C)=O N1(C(C=CC(CC)C)=O)CC(CNC(=O)CCCC2CCC2)(OC)C1 c1(C(N2CC(C)CC(NC(C(C)NC(N)=O)=O)C2)=O)cncc(P(C)(C)=O)c1 CC1CN(c2nc(=N)nc(N3CC4CC3CS4=O)[nH]2)CCC1(F)F c1(C(=O)NCC(CNC(CSc2ccc(C)cc2)=O)F)cc2n(c1)CCOC2 N1(C(CC(C)O)=O)CCCC(NC(c2nnc(S)n2C)=O)C1C CCCC(C(=O)N(C)Cc1nc(Cc2ccccc2)no1)N1CCCC1 C(N=c1cc(CC(C)C)nc[nH]1)C1CCN(C(CCc2ncc(C)[nH]2)=O)CC1C Cc1cc(N)cnc1C(=O)NCCCCC(C)NC(C1(C(C)C)CCCO1)=O n1(CCC)nc(C)cc1C(=O)NC1CCC(CNC(C2(C#N)CC(C)C2)=O)C1 N1(C(C2C(=C)C2)=O)CC(NC(=O)CC2CCS(=O)(=O)C2)CC1C c1(C(C)C)cc(CC(=O)NCC(C)(F)CNC(C2(CF)CC(=O)C2)=O)on1 C(=O)(CC(CN(C)C)CC)N1CCC(N(C(CC)=O)C)C1 C1(CCC=C)(C(=O)NCCCCCN(C)CC)CN(C(=O)COc2ccsn2)C1 Cc1nc(N(C2CC23CCNCC3)C(c2cc(O)no2)=O)c2sccc2n1 N1(C(C(n2cc(C(c3ccccc3)=O)nn2)C)=O)CCN(C(=O)C(C)(C)CF)CC1 C1(CC(N2CCC(NC(CC3CC(CC)C3)=O)(CF)C2)=O)CCCCC1(C)C C(CO)(C(C)NC(=O)C(CO)NC(N)=O)NC(C1(CCC)CCC1)=O c1(C(N2C(CNC(c3cc(CCC)oc3C)=O)CC2)=O)cc2nc[nH]c2cc1F N1(C(c2c(C)nc(C)[nH]2)=O)CC(CNC(C2CCC(C)O2)=O)CC12CCOCC2 CCC(C)CC(=O)NCCCCNC(n1nc(NC)c(Br)c1)=O c1(CC(=O)NCc2cc(OC)c(O)cc2)cnc2ccccc2c1 CC1CCC(CNC(c2cccc(O)c2F)=O)CN1C(c1cnns1)=O c1(C(N2CCC(N(C(=O)Cc3ccc(F)cc3)C)C2)=O)coc2c1CSC2 C1(N(C(c2cc(CC)on2)=O)C)CCC2(CC1)CCN(C(c1csc(=N)[nH]1)=O)C2 C(CC(N)=O)(C(=O)NCCc1nccs1)NC(c1c(CC)n(C)cc1)=O N1(C(C2C(OC)(OC)CC2)=O)CCCC2CN(C(=O)CCF)CCC12 CC(C)C(F)(CN)C(=O)Nc1ccc(Oc2ccccc2F)cc1 Cc1cc(F)cc(C(=O)NC2(CNC(=O)Cc3ncn4c3COCC4)CC2)c1N C#CCCC(O)C(=O)NCC1(CNC(c2cnc(C)nc2C)=O)CC1 c1(C(=O)NCC(CCCC)NC(C2CCCC(O)C2)=O)ccc2c(c1)nnn2C O=C1Cc2cc(CC(=O)NC3CCC(NC(c4cc(Cl)no4)=O)CC3)ccc2N1 c1(C(=O)NC2CC(CNC(=O)C=CC3CCCC3)C2)cc(CO)ccc1Cl C1(CNC(CC2(N(C)C)COC2)=O)CCCN1C(C1(CF)CC1(F)F)=O c1(C(=O)NCC(CCOC)NC(=O)C(C(C)C)N(C)C)occ2c1CCCC2 N1(C(COCC(C)C)=O)C2CCC1CN(C(c1ccno1)=O)CC2 C1(C(=O)NC2CC(N(C)C(c3ccc(CN4CCCC4)o3)=O)C2)CC(F)C(=O)N1 c1(C(N2CCN(C(C3CC(O)C3)=O)CC2CCO)=O)cc2c([nH]1)CCCC2 c1(C(=O)NC(c2c(C(=O)NCC(C)OC)con2)C)cnccc1C CC(CC1CC1)C(=O)N1CC(C(N)=O)(CNC(=O)COc2ccon2)C1 CC1CN(C(=O)C(C)(C)C2CCCN2C(=O)CN2CCCCC2)CCC1O C1(C(N(CC(CC)C)CC)=O)CN(C(c2cc(C)oc2C)=O)CC1(F)F C1(NC(c2c(C)snn2)=O)CC2(CCN(C(=O)C(C)SC(C)C)CC2)C1 CC1(C)CCCCC1CC(=O)NC1(C)CCN(C(c2cc(O)cc(O)n2)=O)C1 C12(C(N3CCCC(C)C3CO)=O)CCC(CC1)N(C(=O)C(O)C1CCCC1)C2 N1(C(c2ccc(N(C)C)cc2)=O)CC(CNC(=O)CCC(F)(F)F)OC(C)(C)C1 C12(CNC(C(CC)CC)=O)CC(COC)(CN1C(c1cc(C3CC3)nn1C)=O)C2 Cc1cc(-n2c3nnc2SC3C)cc(C)c1.C1(CCCCC(=O)O)CCNCC1 CC1(C)CC(S(=O)(=O)N2CC3CC2CC3O)CCN1 C1(Nc2cc(C)ncn2)CN(C(C2CCN2C(C)(C)C)=O)CC1(C)C Cc1ncnc(C)c1CC(=O)NC(C)C(C)NC(=O)COc1ccc(O)cc1 c1(CC(C(=O)O)N(CCN(C)C)CCN(C)C(N)=O)cccc(OC(F)(F)F)c1 C#Cc1cnc(NC2CCN(C(c3ccc(C(C)(C)C)cn3)=O)C(C)C2)nc1 N1(C(C)=O)CC2CN(c3cc(C(F)(F)F)ncc3C#N)CC2C1 Cc1ncnc(C)c1CC(=O)NCC(CO)NC(=O)C(c1cccnc1)C C1(CNC(CSc2cccc(C)c2)=O)COCCN(C(=O)CC#N)C1 c1(NC(C2(C)N(C(C3CCC(=O)NC3)=O)CCC2)=O)ccc2nc(O)[nH]c2c1 N1(C(C(CC)OC)=O)CC2(C1)OC1(CO)CC2(C(=O)OC)C1.C(=O)(CCC)NC1CC1 C1(C(=O)NC2C3(CC(NC(c4ccn(CCCC)n4)=O)C3)C2)CCC2CCC1O2 C=CCC(CCCCC)C(=O)NCC(CC)N(C)C(C12COCC1C2)=O C1(C(N2C(C)CC(N(C(C)=O)Cc3ccccc3)C2)=O)CCc2nnc(O)n2C1 c1(CC(C)C)ccc(C#N)c(NC(C2CCCCN2C(C2CC=CCC2)=O)C)n1 Cc1ccccc1-n1cc(CN(C(=O)CN(C)Cc2ncc[nH]2)C(C)C)nn1 C1(C(=O)OC)(OC)CCN(C(=O)C(N2C3CCC2C(CO)C3)=O)CC1.C(C)C C(=O)(CCCC(N)=O)NCC1N(C(Cc2c(C)nc(C3CC3)s2)=O)CC1 c1(C(=O)NCC2CC(C(=O)NC(c3ccco3)CO)CO2)cnn2c1OCC2 C12(C(=O)NCCOC3CCN(C(c4c(C)nsc4)=O)C3)CC1Cc1c[nH]nc12 Cc1nc2cc(O)nn2c(C)c1CC(=O)NCC1(O)CN(C(=O)COCCF)C1 Cc1cc(C)c(C(=O)NC2COCC2NC(C2(F)CCCN(C)C2)=O)c(C)n1 C(=O)(CS(=O)(=O)C(C)(C)C)NCC(C)CN(C(=O)CC1CC1C1CC1)C N1(C(Cc2cnc(C)s2)=O)CC2CC1CN2C(c1snc(C)c1N)=O N1(CC)C(=O)CCC1CC(N1CCCCC1CN(C)C(C1CN(C(C)=O)C1)=O)=O N1(C(c2cc(OC)ncc2)=O)CC=C(C(=O)N(C(C)CCSC)C)C1 C(CC(C)(O)C(=O)N1CC(C(=O)NC2CCOCC2F)C(F)(F)C1)N(C)C C1(C(=O)NCCCN(C(=O)C(C)=C(C)C)CC)CCC(=O)CC1C C1(NC(C(C(CNC(C2(C(C)C)COC2)=O)C)F)=O)CC2C(O)C(O)CC12 C1(CC(=O)NC2CN(C(CCC=C=C)=O)CC2C)CCCC(F)(F)C1 C1(CNC(c2ccc(OCCC)cc2C)=O)CCOCC12CCC2 C1(CC(=O)OCC)(CC(=O)NCCNC(=O)C(C)Oc2cccnc2)CCCC1 C1(C(=O)NC2C(C)(C)C(CC(=O)NCCC(N)=O)C2)CC(=O)NC(=O)C1 c1(C(=O)NCC(C)NC(C(c2ccc(C)cc2)C(C)C)=O)nc2ncccn2n1 c1(C(N2CC3C(C2)N3C(C2(c3cccs3)CC2)=O)=O)ccc(Br)c2ncccc12 c1(C(=O)NCCCCCN(C(CCN(CCC)C)=O)C)sc2ncccc2c1N c1(CNCC2(C(=O)NCc3cc(C)no3)CC2)cncc(C#N)c1 c1(C(N(C2CCN(C(c3nc(C4CCC4)co3)=O)C2)C)=O)ccc(OC2CC2)cc1 Cc1cccc(Cl)c1CC(=O)NCC(C(C)C)NC(=O)CCCCF N1(C(C(C(CC)O)C)=O)CCOC2(CCN(C(c3ccnc(Cl)c3N)=O)C2)C1 C1(NC(c2cncnc2)=O)CC(CNC(c2cc(C3CC3)ccn2)=O)C12CCC2 CCC(CC(=O)N1CCN(C(=O)Cn2cc(Cl)cn2)C(C)C1C)CC(C)C N1(C(C)=O)C2CCC1CC(NC(=O)C(c1ccc(Cl)c(Br)c1)(F)F)C2 CCC(CNC(c1cc(OC)ccn1)=O)N=c1cc(C2CC2)nc(Cl)[nH]1 c1(C(N2CC(C(C)NC(=O)CC3C=CCCC3)C2)=O)n[nH]c2cc(OC)ccc12 c1(N(CC(C)C)C)ccc(C(=O)NC2CCCC2NC(=O)Cn2cncn2)cn1 C1(C(C)NC(CCNS(CC)(=O)=O)=O)CCN(C(=O)CC2(O)CCCOC2)CC1 c1(C)cc([N+](=O)[O-])ccc1F.c1(O)cncnc1N(C(C1CCCNC1)C)CC C(=O)(CC(C)C(C)(C)NC(=O)C(COC)OC)N(CC(CC)OC)C C(=O)(C(C(C)C)NC(=O)C(CNC(=O)C(=O)NCC1CC1)CSC)OC C1(NC(C2CCCN(c3nccs3)C2)=O)CN(C(=O)C2=CCC2)CC12CC2 C(=O)(C(F)(F)C(F)(F)F)NCC1(F)CCN(C(c2ccc(OC)c(N)n2)=O)C1 N1(C(Cc2c(C)oc(C(F)(F)F)n2)=O)CCN(C(C2(C3CC3)CC2)=O)CCC1C c1(CCC)noc(CCCC(=O)NCC(CO)NC(c2cc[nH]c2)=O)n1 C1(C)(C(=O)NCC2CC3CC(NC(=O)OC(C)(C)C)C3C2)CC(C(C)C)=NO1 c1(C(N(C(CN(C(C(C)C2CC2)=O)C)C)C)=O)ccccc1C(F)(F)F C(=O)(C1=CCCCC1C)NC(CC=C)CC(=O)NC(c1nc(C)no1)C CC1CCCCN1CCNC(=O)CCCNC(c1cnn[nH]1)=O N1(C(CCCN(C(=O)OC)C)=O)CCC(CC(N)=O)(NC(C2CCSC2)=O)CC1 N1(C(CCC=C)=O)CCC(O)(CCNC(C2(COC)CCCO2)=O)C1 C(=O)(CCC(C)CN(C)C)NC(C)CNC(c1cnn(-c2ccccc2)c1F)=O N1(CC(=O)N(CC(C)NC(C2(CCF)CCC2)=O)C)CCCC(C(F)(F)F)C1=O CC1CN(C(c2cnn(CCNC(C3(O)CCC3)=O)c2)=O)CC(=O)N1C C#CCC(CC(=O)N1CCOC2CC12)NC(=O)C(=O)C(C)CC Cc1cccc(C(=O)NC2CN(Cc3cccnc3)CC2F)c1C c1(C(C)=O)cc(C(N2CC=CC2C(=O)NCC2COCC2O)=O)no1 N1(C(C(CCCC)C)=O)CCC(C)(C)C(CNC(c2cnn3ccn(C)c23)=O)C1 c1(C(=O)NCCCCCCn2cc(CCOC)nn2)cccc2ccn(C)c12 C1(NC(COC(CC)(C)C)=O)(CC)CCN(C(=O)CCCc2csc(C)n2)CC1 c1(NC(c2cccc(Nc3nc(Cl)ncc3F)c2)=O)ccc2c(c1)OCO2 N1(C(CCCOCCC)=O)CCC(CC(N2CCC(C)(C)C2C)=O)C1(C)C C1(CNC(Cc2c(C)noc2C)=O)COCCN(C(c2ccc(N)cc2O)=O)C1 N1(C(CCCNC(=O)CNC(=O)C(C)(C)C)=O)CC2(CCOCC)CCC1CC2 C1(NC(C(CC)SC)=O)CCN(C)C1(C)C.C12CC(C1)NC2=O c1(C(N2CC3(CCN(C(C(C4CCC4)OC)=O)C3)C2)=O)cnc2ncnn2c1N C12(C(=O)NCCc3n(C)cnn3)CCN(C(C3CC4CC(=O)C3O4)=O)CCC1C2 N1(C(CCc2n(C)ccn2)=O)CCC(F)(CNC(=O)Cn2cnnc2O)C1 c1(C(N2C(CCC)(C(=O)OC)CCC2)=O)cc2nc(C)cc(C(F)(F)F)n2n1 c1(C(=O)OC(C)(C)C)coc(COCC(C)NC(C2CC(F)(CNC)C2)=O)c1 CC1CCN(C(C2CC3(CSC3)C2)=O)CC1NC(c1ccnc(CO)c1)=O N1(C(C23N(C(CCSCCC)=O)CCC2C3)=O)CC2(CC2)CC1CO N1(C(C2CCC(=O)N2)=O)CC2(CC(NC(c3ncccc3Br)=O)CO2)C1 Cc1ccc2c(c1)CC(C(=O)NCC(C)N(C(=O)C1=NOC(C)C1)C)S2 c1(OC)nc(C)ccc1C(C(=O)NC1CC(F)(F)C1)N(C)Cc1cnc(C)s1 CCCCC(C(=O)NC(c1cn(C)nn1)C(=O)NC1CN(C)CC1O)ON=C(C)C C1(CNC(=O)Cc2ccncc2)CC2OCCC2N1C(=O)CCc1ccccc1 c1(NC(CC2(C)CN(C(c3ccc(Br)c(O)c3)=O)C2)=O)cccc(Cl)c1Br c1(OC)cc(C(N2CC3CC(CNC(C4CC4CF)=O)C3C2)=O)cc(N)c1OC C(=O)(C1OCCc2ccccc21)N(C(C)CNC(C12CC(C)(C1)OC2(C)C)=O)C c1(C(N2C(Cn3cc(C(C=C)(C)O)nn3)CC2)=O)cnc(O)cc1OCC N1(C(c2nc(C(C)OC)oc2)=O)CCC(C2(C)CC2)CC1 c1(CN(C2(CO)CCOCC2)C(C(C)N)=O)cccc(C(F)(F)F)c1.COC Cc1c(F)ccc(C(=O)NCC2(CO)CCCN(C(C3(C)CCCO3)=O)C2)c1N N1(C(C=C(COC)C)=O)CCN(C(c2cc(-c3ccoc3)[nH]n2)=O)C2CCC12 c1(C(=O)NCC(CNC(CN(C(C)C)C)=O)CO)c(Cl)ccc(F)c1N c1(CC)cc(NC2CC(c3ncc[nH]3)C2)nc2ccccc12 N1(C(=O)NCCCl)CC2CCN(Cc3ccc(I)cc3O)CC2C1 CC(C)(CC(F)C(=O)NC1CC2C=CC1C2)NC(=O)CCCN=[N+]=[N-] C1(CNC(C(C(C)C)C#N)=O)COC(C)(C)CN1C(=O)Cc1csc(Cl)c1 C1(COC(C(CC)(C)Nc2nc(NC)cc(C)n2)C2CC2)CCc2cnn(C)c2C1 C1(NC(C#CC2(C)CC2)=O)CCC2(CC1)CCN(C(C1CCS(=O)(=O)CC1)=O)C2 C(=O)(C1CCc2cccc(O)c21)NC1CN(C(C(C)OCCC(C)C)=O)C(C)C1 c1(C(N2CC(C)CC(NC(CN(CC)CC)=O)C2)=O)cc2cccc(F)c2s1 CON=CC(=O)NCC(C1CCCCC1)NC(=O)CC1OCCC1C c1(C(CO)NC(C(=O)NC2CC(C#C)C2)=O)cccc(F)c1 C(=O)(CCCC(C)(F)F)N(C1CN(C(c2cc(O)ccc2Cl)=O)CC1F)C N(C(=NCCC1CCCOC1)NC1CCC1)CC(CC)(C)C C1(NC(CSCC#C)=O)(CNC(C2CCCOCC2)=O)CCCCCC1 C1(C(N(OCC)CC)=O)CCC(C)(C)N(C(C2CC23CCCCC3)=O)C1 C1(NC(CCC#CC)=O)C2CC3CN(C(=O)Cc4cc(C)cc(F)c4)C1C3C2 C1(CNC(=O)C(O)C2CCCC2)CN(c2ncnc3sccc23)CCC1(F)F CC(C)C(C(=O)N1CC(NC(=O)Cc2ccc(Cl)nc2)CC1CO)C1CCC1 C1(CNC(C(C2CN(C(c3cn(C(C)C)nn3)=O)C2)OC)=O)CCOC1(C)C N1(C(C(C)SCC)=O)CCN(C(c2ccc(O)cc2C(F)F)=O)CC1CO n1(CC(=O)NC(Cc2ccccc2)C2CC2)cc(Br)cc(Cl)c1=O N1(C(C=Cc2occ(C)n2)=O)CC(C2CN(C(c3ncc4[nH]ncc4n3)=O)C2)C1 c1(C(=O)OC)c(C)sc2cc(C(=O)NC(CO)C(C)NC(=O)CC(C)C)[nH]c12 C(=O)(CCCNC(c1nccn1C)=O)N(CC(F)F)CCOC C1(C(N2CC=CC(NC(CN(C(COC)=O)C)=O)C2)=O)CCCN(S(N)(=O)=O)C1 C(=O)(CC1COc2cc(O)ccc21)NC1(CNC(C2C(C)C2(F)F)=O)CCC1 c1(C(=O)NC2(CNC(=O)CN3CCCCC3)CCC2)ccnc2nccnc12 c1(C(N2CC(OC)(CNC(C3CCC4CCC34)=O)C2)=O)ccc2c(c1)CCCN2 C(=O)(C(COC)CC)NCCN(C(c1c(CC)cc[nH]1)=O)CC1CC1 C1(C(=O)NCC=C2CCN(C(c3ccncc3F)=O)CC2)CCc2cncn2C1 CC1CC(NC(=O)C=C(Cl)Cl)CN(C(C2CC(C3CC3)=NO2)=O)C1 c1(C2(C(=O)NCC(CC=C)NC(=O)CC(C)C3CC3)CC2)ccnc(Cl)c1 C1(C(N(C)CC2(NC(=O)C=CSc3ccccc3)CC2)=O)CC2CCC1C2 Cc1cc(C(=O)NCC2(C)CCCN2C(=O)COc2ccc(Cl)cc2)cc(O)n1 C1(NC(C2C(C)=CCS2)=O)CCN(CCNC(=O)Cc2nc[nH]n2)CC1 C(C(=O)N(C)Cc1ccn(CC)n1)(C(C)CC)N(C(COCCC#C)=O)C N1(C(c2cc(C)sc2)=O)CCC2(CCC2)C(CNC(c2cc(F)cc(F)c2)=O)C1 c1(C(=O)NC2CCN(C(C3(C(C)C)CC3)=O)CC2F)cc2cccnc2[nH]1 c1(OCC)ccc(C(=O)NCC(C)(C)CNC(=O)CC23COC(C2)C3)cc1 C1(C#N)(CNC(CC2C(C(=O)NC3(CC#C)CCOC3)CCC2)=O)CCOCC1 C(C(CC(C)C)C(=O)NCCNC(C1(CO)CCCCC1)=O)OC c1(C(N2C(C)CC(CNC(CCC=CC)=O)C2)=O)cccn(C2CCC2)c1=O C=CCC(CC)C(=O)NCC(C)CNC(=O)CSc1ccccc1C N1(C(c2ccc(CSC)o2)=O)CC2CC(NC(c3coc(C)n3)=O)C2C1 N1(C(C2CC(OC)C2)=O)CCN(C(C2CCC(=O)NC2)=O)CC1c1nccn1C N1(C(C2CNC(=O)N2)=O)CCC(CO)(NC(=O)CCC2NC(=O)NC2=O)CC1 CCCC(CCC)C(=O)NC1CCCC12CN(C(=O)C(CC)c1ccccc1)C2 N1(CCN(C(C=C(CCC)C)=O)C)CCN(C(C2CCC(C(N)=O)C2)=O)CC1 CCC(CN(C)C)CC(=O)N1CC(CO)(NC(c2cccc(CO)c2C)=O)C1 c1(C(N2C(C(=O)Nc3n(C(COC)C)ccn3)CC2)=O)ccc(OC)c(O)c1 CS(=O)(=O)c1ccc(OCC(=O)NC(=O)Nc2ccccc2)cc1Cl N1(C(CCC(=O)NC)=O)CCCCCC1C(=O)NC1CCC2CCC12 CCC(CCC(=O)N(C1CC2CCC1O2)C)NC(=O)C=Cc1nccs1 C1(C(=O)NC2(c3ccc(F)cc3)CCN(C(=O)CO)CC2)Cc2cccnc2C1 N1(C(N(C)Cc2c(OC)cccc2)=O)CCN(c2ccc(F)cn2)CC1C c1(C(=O)NC2C=CC(CNC(c3cscc3Br)=O)C2)cc2n(n1)CCCC2 C(=O)(C(C)CCCC(C)=O)N(C(C(N1CC(C#C)C(OC)C1)=O)(C)C1CC1)C C#CCC(C)(C)C(=O)NCC1(CNC(c2c[nH]nc2CC)=O)CC12CCC2 c1(C(N2CCC(NC(CC(C(C)C)O)=O)(CO)C2)=O)cnc2[nH]nc(O)c2c1 C1(NC(C(C)N(C(C2C3CCC(C3)C2C)=O)CC)=O)CN(C)C(=O)C12CC2 C(=O)(N=c1ccc(C2CC2)n[nH]1)Nc1c(CC)nc(CNC(=O)OC(C)(C)C)o1 C1(NC(C2CN(C(C)C)C(=O)C2)=O)CCN(C(=O)Cc2cncs2)CC1O C1(C)(C(=O)NC2CC(C)(NC(C(C)N(C(C)=O)C)=O)C2)CCOC(C)C1 c1(CCCSCC)cn(C2CCN(C(=O)C(C)(C)C)C2)nn1 C1(C(=O)NCc2ncc(C)s2)CC(F)(F)CN1Cc1cnc(Cl)cc1Br C(C(CC(C)C)C(=O)N1CCCCC1CN(C)C(C1CN(C(C)=O)C1)=O)OC Cc1cccc(C(=O)NC2CC(CO)N(C(=O)Cn3cnccc3=O)C2)c1Cl C1(CC(C)C)(C(=O)N(C)CCN(C)C(C2CCCN2C(C)C)=O)CCNC1=O Cc1nc(O)ccc1C(=O)NCC(CC1CC1)C(=O)NCC1(C2CC2)CCC1 N1(C(C2C(OCC)CC2)=O)CCOC2(C1)CN(C(=O)CSCc1ncnn1C)C2 Cc1cnc(C(C)NC(c2cc(C3CC3)ns2)c2nnnn2CC2CC2)s1 c1(CC(N2CCC(O)(CNC(C3(CC)CC3)=O)C2)=O)cc(F)c(C)cc1F CCCCC(C)CCC(=O)NC1C2CC(NC(c3csc(C4CC4)n3)=O)CC12 c1(C(N2CCC(NC(c3occ4c3CCC4)=O)C2)=O)ccc(Cl)c2cccnc12 c1(C(=O)NCCCOc2c(C)cccc2C)nccc2c1n(C)c(=O)n2C C1(NC(c2c(CN(C)C)cccc2)=O)CN(C(C2(C)CCCS2)=O)CC(F)(F)C1 C1(C(=O)NC(C(=O)OCCC)C)CN(C(C2(F)CCC2)=O)CCO1 c1(OCC)cnc(C(=O)NCCN(C(c2ncn(CC)n2)=O)CCOC)c(Cl)c1 n1(CC)nc(C(N2CCCCC2CNC(=O)C(F)(F)CC2CC2)=O)cc1C C=C1CC2CCCC(C1)N2C(C1CN(C(=O)C(C)OCCOC)CC1(F)F)=O N1(CC2CCC(C)(C)C2)C(=O)CN(CCP(C)(C)=O)C1=O C(=O)(C1CCCc2sc(=N)[nH]c21)NCCNC(C1(C)CC1(F)F)=O CC1CCN(C(=O)Cc2cncnc2)C1CNC(c1ccc(-c2ccco2)s1)=O N1(C(c2cccc(OCC(C)C)c2)=O)CCC(NC(=O)C2=CCCS2)C12CCC2 c1(OCC=C)cccnc1C(N1CCCC1CNC(=O)CCNS(C)(=O)=O)=O C1(CCOC)CN(C(c2nnc(Cl)cc2N)=O)CCN1C(C1CN(C)CCO1)=O CCS(=O)(=O)C1(CNC(N2CCC(NS(=O)(=O)c3cccs3)CC2)=O)CC1 Cc1nc2cc(C(=O)NCC3(C)CC(NC(C4CC=CCC4)=O)C3)cnc2s1 C1(CNC(c2cnc(CC)o2)=O)CCCCN(C(c2ccc(C)nc2C)=O)C1 c1(C(C(N2CCC(N(C(=O)Cc3cscn3)CC)C2)=O)(F)F)ccc(C)cc1 C1(N(C(C(CC)c2ccccc2)=O)CC)CCCN(C(=O)C(O)CCSC)C1 CCCCCCCC(F)C(=O)NC(C)(CNC(c1conc1C)=O)CO N1(C(C(C)NC(=O)CCNC(=O)CO)=O)CCC2(CCSC2)C1 N1(C(=O)OC)CCCC(N=c2[nH]c3c(c(=NCCc4ccsc4Br)[nH]2)SCC3)C1 N1(C(c2n[nH]c(C)c2F)=O)CCC2(CCCN(C(=O)CN3CCN(C)CC3)C2)C1 N1(C(CN(C)S(N)(=O)=O)=O)CCC(CNC(=O)C2=CCCCO2)C(F)(F)C1 N1(C(c2c(C)nc(O)cc2)=O)CCCC(C)(C)C1CNC(C1(C(N)=O)CCC1)=O c1(OCCC)cccc(C(=O)N(CC(C)(C)NC(C2CC2CCOC)=O)C)c1 c1(NC(CN2C3CC(C(=O)NCC)C2CC3)=O)nc2ccc(OC(C)C)nc2s1 c1(C(=O)NC(CN(C(CC2N(CC)CCC2)=O)C)C)ccc(F)cc1C1CC1 C1(CNC(C2CC2F)=O)CCCC12CCN(C(=O)CC1CSCCS1)CC2 Cc1ccc2c(c1)SC(C(=O)NC1CC(NC(c3coc(O)n3)=O)CC1O)C2 C(=O)(CC(C)CC(C)(C)C)NC1CN(C(c2cc(OC)cc(C)c2N)=O)C(C)C1 N1(C(C(C)SCC)=O)CC(SC)(NC(CC2(C(=O)NC3CC3)CC2)=O)C1 N1(C(C(CC)(C)CNC(=O)C(F)F)=O)CCC2CC1C(=O)O2 N1(C(C2CCC(CC)O2)=O)CCCC12CCN(C(=O)CCC(=O)OC)C2 c1(CNC(c2n(C(CC)C)nnn2)c2coc(C)n2)cccc(Br)c1 S(=O)(=O)(c1ccc(NCC(F)C2CCC2)c(C#N)c1)NCc1c(CC)nn(C)c1 c1(CC(=O)NCCC2(OC)CN(C(c3sc(CO)nc3C)=O)C2)ccc(C)cc1 N1(C(c2n(C)c(S)nc2)=O)CCC(C2(NC(=O)CC3CC=CCC3)CC2)CC1 Cc1ncn(C)c1C(=O)NC(C)C(C(C)C)NC(c1cnn(C2CC2)c1C)=O N1(C(c2cc(C)ns2)=O)CC(CNC(=O)CSCc2csc(=N)[nH]2)CCC1C N1(C(c2c(C)n[nH]c2C)=O)CCC2(CC2NC(C2CC(C)C2)=O)C1 C1(CNC(C(C2CCCCCC2)C)=O)CN(C(c2ccccc2)=O)CC1O C1(NC(c2ccn(CCNC(C(CC=C)C)=O)c2)=O)CCc2nncn2C1 C(=O)(C(C)CC(C)C(C)=O)NC1C(CC)N(C(c2cn(C)nc2OC)=O)CCC1 c1(CC)cnc(NC(=O)C(=O)NCC2CSCCS2)s1 N1(C(C2ON=C(C)C2)=O)CC2(CC(C(=O)NCCc3csnn3)CO2)C1 C1(NC(c2c(CC)oc(C)c2)=O)CC(C(=O)N(C)Cc2ccc(C)cc2)=CC1O C1(NC(CCSC)=O)CC=CCC1C(=O)NCCn1cnc(CO)c1 C(=O)(C(CC)N(C(=O)Cn1cc(COC)cn1)C)NCC(=O)N(C)CC S(=O)(=O)(c1ccc2occc2c1)NCC1C=CCN(C(=O)Nc2ccccc2)C1 c1(SC)cccnc1Cn1ccnc1Cc1ccccc1 N1(CCC)CCN(C(C2CCC(c3cccc(Cl)c3)C2)=O)CC1 C(=O)(CC(O)CNC(C1CC(C)=NO1)=O)NC(C(=O)OCC)C C1(CNC(c2cn(CC)nc2)=O)CCC(C(N2CCC2C(C)C)=O)CC1 c1(C(=O)NCCCNC(c2c(N)ccc(C(C)=O)c2)=O)cc(S(N)(=O)=O)sc1C c1(OC)cc(OC)c(NC(C2CN(C(=O)CCc3ccc(C)s3)CCN2)=O)cn1 C(C(C)(C)C(C)(C)C)NC(C(c1ccccc1)NC(Cn1ncn(C)c1=O)=O)=O c1(C(=O)NCCC(C)NC(c2c(COC)cccn2)=O)oc2ccccc2c1C Cn1nnnc1SCC(=O)NC1(CCNC(C2CC2C(F)F)=O)CC1 c1(C(N(CCN(C(C(CC=C)NC(C)=O)=O)C)C(C)C)=O)ccc(OC)nc1C CCCCC(CC)C(=O)NCCCOCCN(C)C(C1CSCCS1)=O C(CS(=O)(=O)CC(=O)N1CCN(C(c2cnn(C)c(=O)c2)=O)CC1C(C)C)OC c1(C(=O)NCC(CNC(c2ccnn2C)=O)OC)cc(Cl)cc(F)c1N c1(CN=C(NCC2(C)COCCO2)NC2CC2)cc2c(cc1Br)OCCO2 N1(C(C2NC(=O)OCC2)=O)CCC2(CCC2)C(CNC(C2(CO)CCCC2)=O)C1 C#Cc1ccc(Cl)c(C(=O)NC(C)C(C)NC(c2cc(C(C)(C)C)nn2C)=O)c1 Cc1cc(F)ncc1C(=O)NC(C1CCN(C(=O)CCc2cccs2)C1)C c1(C(C)C)sc(Cl)nc1CN1CCN(C2CN(C(=O)C(C)(C)OC3CC3)C2)CC1 C(C(F)(F)C(F)(F)F)c1n(-c2ccc(C(C)N(C)C)cc2)nc(C2CCOC2)n1 Cc1cc(Cl)cc(N)c1C(=O)NC1CN(C(=O)CN2CCC2C)C(C)(C)C1 C1(NC(C(c2ccccc2)C)=O)CC2CN(C(=O)CCCCC3CC3)CC12 Cc1ccc(C(F)(F)C(=O)NC2CCC2NC(c2cc(C)ncn2)=O)nc1 c1(C(N2CCC(C)C(NC(C3(F)CCCC3)=O)C2)=O)cc2ccccc2o1 C(CSc1cn(C(C)(C)C)nn1)(CO)(CO)N(C(c1[nH]cc(C(C)=O)c1)=O)C C1(NC(=O)NC(C(F)(F)CO)C2CC2)CCn2nncc2C1 C1(NC(C(C)CC(F)(F)F)=O)CCCCC12CCN(C(C1CC3CCC1O3)=O)C2 C1(CNC(=O)Cn2ncnn2)CN(C(C2CC3CCC2CC3)=O)CCC12CCC2 Cc1cccc(Br)c1C(N1CCC(=CCNC(c2cccnc2Cl)=O)CC1)=O C1(CNC(c2ccc(F)s2)=O)CC2(CCN(C(c3cc[nH]c3C3CC3)=O)C2)CO1 N1(C(c2ccc(F)c(CO)c2)=O)CC2CCCN(C(C3C4CCC3CC4)=O)C2C1 C(=O)(C1CCCn2nccc21)N1CCCCC(N(C(=O)C2=C(Cl)CC2)C)C1 c1(C(=O)NC2C3CN(C(c4ccccc4O)=O)CC32)c(O)ncc2c1CCC2 C1(NC(c2ccc(C)cc2Cl)=O)CN(C(=O)CC2CCCC(=O)N2)CCC1(C)C c1(C(=O)NC(CC)CNC(c2cncc(F)c2Cl)=O)ccn(C)c(=O)c1O Cc1ccnnc1C(=O)N(C1CCN(C(=O)Cc2ccccc2F)C1)C N1(CC(=O)OCCCF)CCCC(CC(F)F)C1 c1(C(N2CCN(C3CCN(C(=O)COC4CCC4)C3)CC2)=O)cc([N+](=O)[O-])c[nH]1 c1(N(C)C)ccc2cc(C(N3CCN(Cc4cncs4)CC3)=O)ccc2c1 CCCCC(O)C(=O)NCC(O)CN(C(=O)C(C)(C)COCC(F)F)C C1(NC(=O)CCC2CCC2)CC2CCC1CC2NC(C1CC2CCCCC2O1)=O c1(OC)ccc(Cl)c(C(=O)NCCC2CCN(C(=O)C3=COCC3)C(C)C2)c1 c1(C(N2C(C)(CNC(c3nn(C)c(Cl)c3)=O)CCC2)=O)c[nH]c2cccc(F)c12 c1(C(=O)NCC2CCC(C(=O)NCc3cc(CC)no3)C2)cc(C)n(C)c1 c1(NCc2ccc(C)cc2Br)ccc(S(=O)(=O)NCc2ccn(C)n2)cc1Cl Cc1cc(NC(=O)CNC2CCN2C(=O)CCNC2CC3(CC3)CO2)ccc1N n1(CC(=O)OC)cnc(C)c1C(=O)NCC1CC1CNC(c1oc(C)nc1C)=O CCCC(C(O)C(=O)NCc1cncc(F)c1)NC(=O)C(C)CCOC C(=O)(C(O)C(C)C)NCCOCCNC(c1n(CCC)ccc1)=O N1(C(CCNC(C)=O)=O)CCC(C(N2CCN(CCCO)CC2)=O)C(O)C1 CC(CO)(CO)C(=O)NC1CCC(C(=O)Nc2cc(F)cnc2Cl)C1 O=C1OCc2c(C(=O)OCCC(=O)NC3CCCCC3)cccc21 N1(C(C2COC(C)(C)OC2)C(=O)NCC(=O)OC)CCCC(C)C1c1cccs1 CN1CCOCC1C(=O)NC1CCC(C(=O)NOCC2(F)CCC2)C1 Cc1nc(C)n(-c2ccc(C(=O)NC(C)(C)CNC(C3(C(F)F)CC3)=O)cc2)n1 c1(C(N2CCC(NC(CC3ON=C(C)C3)=O)(CF)C2)=O)ccc(Cl)c(C)c1N CCC(O)C(F)(F)C(=O)NC1CCN(C(=O)C=Cc2ccccc2)C(C)C1 c1(OC)ccncc1CNC(=O)C(C)CN(C)C(C1CCSC1)=O C1(F)(CNC(C2C=CCC2)=O)COCCN(C(=O)CC2CCCCC2)C1 c1(C(N(CCN(C)C(c2cc(Cl)n(C)n2)=O)C)=O)cc(O)nc2ccc(Cl)cc12 C(=O)(C(CC#CC)NC(c1ccc(C)cc1O)=O)NC(CCC=C)(C)C C1(C(=O)NCC(C)O)COCCN(CC(O)CN2CCOCC2)C1 CC1(C)OC(=O)CC1C(N1CCOCCC1C(=O)NC1CCS(=O)CC1)=O c1(C(N2CC(CNC(c3cnc(C)s3)=O)C3(C2)CC3)=O)cc2cccnn2n1 C1(NC(C2(SCC)CC2)=O)COC2(CCN(C(=O)CCC3CCC3)C2)C1 c1(C(=O)NC2C(CNC(c3ccc(CCC)cc3)=O)C2)cccc2c(C)[nH]nc12 N1(C(c2cn(CCNC(C3C(C)(C)C3(C)C)=O)nn2)=O)CCOCC(C(=O)O)C1 Cc1cnc2c(C(=O)NC3CN(C(C4Cc5cc(F)ccc5O4)=O)C3)cnn2c1 C=CCC(CC)C(=O)NC(c1cccnc1)C(=O)Nc1cnccc1OC C(=O)(C(CC(C)C)CC(C)C)N(CCCCCNC(Cc1ncc(C)o1)=O)C Cc1c(C(=O)NCCN(CC(C)O)C(c2coc(Cl)n2)=O)oc2ccc(Cl)cc12 c1(C(=O)NCC(CNC(CCCCOC)=O)O)ccc(=O)n(C(C)C)c1 C1(C(=O)NC(CN(C(c2c(C(C)C)[nH]cc2)=O)C)C)CC2(C1)CC1(CC1)C2 C(=O)(C1=NOC(C)C1)NC(C(=O)NCC1ON=C(CC)C1)Cc1ccoc1 N1(C(c2c(CC)onc2C)C(=O)NCC2CCCO2)CCc2ccccc21 S(=O)(=O)(c1[nH]c(=NCC2(C)CCOC2)ccc1Br)N1C2CC(OC)C2CC1 C(=O)(C1CCc2ccc(Cl)nc21)NC1C(CNC(C2=C(C)OCC2)=O)CC1 Cc1sc(O)nc1C(=O)NCC(=O)NC1CC=CCC1C(N1CCOCC1)=O Cn1cc2c(C(=O)NCC3C4CN(C(c5ns[nH]c5=O)=O)CC34)cccc2n1 c1(C(=O)NC2CN(Cc3cc(OC)cc(O)c3)CC2(F)F)cc(Cl)cc(Cl)c1O C1(C(=O)NC(CC#C)CO)CC(C)CN1C(=O)COC1CCOCC1 C(c1cccnc1)=CC(=O)NCC(CO)NC(CCn1ncc(C)c1)=O c1(C(=O)NCC(CC)(C)NC(c2cc3ccccc3[nH]2)=O)cccc2nonc12 C1(C(=O)NC2CCN(C(c3ccn(C)c3)=O)C2)CC2C=CC1C21CC1 c1(C(=O)Nc2c(=N)[nH]n(-c3ccccc3)c2)c(F)ccc([N+](=O)[O-])c1F C1(C(=O)NC(C(=O)NCCC(=O)NCC#C)(C)C)CCCNC1=O CC1(C(N2CCC2)=O)CCCN(C(=O)CCCC2CCC(C(=O)O)O2)C1 C#Cc1cc(C(=O)NC2COCC2NC(=O)Cc2ccc(O)nc2)cc(F)c1 N1(C(c2nc(CC)oc2)=O)CCC(NC(c2cc(CC)cnc2OC)=O)C(F)C1 CC(C)CCC(O)C(=O)NCC12CCC(NC(C3SCCCS3)=O)(CO1)C2 N1(C(C(CC=C)(C)N(C)C)=O)CC2CCC1CN2C(=O)C(CC)OC N1(S(=O)(=O)C2CC3CC2C3)CC(O)CC2CCCCC12 C1(NC(CC2N(CC)CCC2)=O)CCOC2(CCN(C(=O)C=C3CCC3)CC2)C1 O=C(N1CCCc2nccnc21)C1(Nc2ccc(Cl)cc2)CCCC1 c1(C(=O)NCC2OCCCN(C(CC(C)C)=O)C2)cnc2cnccc2c1 C1(NC(c2cccc(C(C)C)c2)=O)CCN(C(=O)C(F)CC2CCC2)C1(C)C Cc1cc2ccc(C(=O)NC3CC(C)(NC(c4ccc(F)cc4)=O)C3)cc2[nH]1 c1(N(CC(C)CNC(c2ccsc2)=O)C)cc(-c2ccccc2)ncn1 c1(C(=O)Nc2ccc(NC(CC(C)C)=O)c(F)c2)ccc([N+](=O)[O-])cc1Br c1(OC)ccc(Cl)c(C(=O)NCCCCCCN(C)C(c2ccns2)=O)n1 CCC(CC(C)C)C(=O)N1CCC(CN(c2nccc(C#N)n2)C)C1 c1(C(=O)NC2CCCC(C(=O)NC3(C)C(C)(C)C3)C2)cnc2cccnn12 n1(CCC(=O)NCC2CC2NC(c2ncncc2Cl)=O)cnc2sccc2c1=O C1(CC)CC(NCC2CCC(F)(F)C2)CCN1C(=O)OC(C)(C)C C1(CNC(CC)=O)CCCN(C(c2cccc(-c3ccccc3Br)c2)=O)C1 CC1CN(C(=O)CC(=O)NC2CC2)CCN1C(=O)Cc1cn(C)nc1Cl c1(C(c2n(CC(=C)C)nnn2)NC(C2CC(F)(F)C2)CCC)ncc(Cl)cc1Br N1(C(CCNC(N)=O)=O)CCN(C(=O)CC(F)(F)Cl)CC1CC(F)(F)F C#Cc1cc(NC(=O)CN2CCN(C(c3ccco3)=O)CC2)ccc1C C1(C2CCN(C(c3nc(C(C)(F)F)cs3)=O)C2)(NC(c2ccc(C)nc2)=O)CC1 c1(N2CCC(Br)=C(C)C2)nc(N2CCOC(CC(C)(C)C)C2)nc2cccnc12 CC1CCC(C(=O)NCC=CCl)CN1C(=O)Cc1cccnc1O C1(NC(C2CSCCS2)=O)CN(C(c2ncncc2Cl)=O)CCC1CO C(=O)(C(CC(C)C)OC)N1CC(CCC=C)(C(=O)NCCC=CC=C)C1 N1(C(c2cc(OCC)n[nH]2)=O)CC2CC1CCN2C(=O)CC1=CCCCC1 C1(C)(CC)C=C(C(=O)N(CCNC(c2ccc[n+]([O-])c2)=O)C2CC2)C1 C1(C(N2CCN(C(C(C)=CC)=O)C(CC(F)(F)F)C2)=O)CC2(C1)NC(=O)NC2=O Cc1cc(NC(=O)CCC2CCCN2C(=O)C(C)S(N)(=O)=O)cc(C)c1F C1(NC(c2cc(C(F)F)[nH]n2)=O)CCCC(NC(C2(N3CCOC3=O)CC2)=O)C1 N1(C(CC2CC(OC)C2)=O)CCCCC(CNC(c2cc(Cl)ccc2C)=O)C1 C(C(CNC1(c2nc(C)no2)CC1)CC1CCCCC1)NC(=O)OCC C1(NC(C2(CCC)CC2)=O)CCCC(NC(c2ccccc2SCCO)=O)C1 C(=O)(CC(F)(F)C(F)F)N1CC(OC(=O)Cc2sccc2COC(C)=O)C(F)C1 C1(NC(C2(CC)CC2)=O)CCCCCN(C(c2cc(F)c(Br)cc2N)=O)C1 c1(C(N2C(C)CCN(C(C(C)C3CCC3)=O)CC2)=O)cc(F)c(F)c(N)c1Cl n1(CC)ncc(C#N)c1NC(C1CC1NC(C1CCCC(N(C)C)C1)=O)=O c1(C(N2CC(NC(CC3(C)CCC3)=O)C2)=O)cccn2nncc12 S(=O)(=O)(c1cncc(Cl)c1)Nc1c(C#N)nc(Cl)cc1 c1(C(N2CCN(CC(C)O)CC2)=O)cnc2ccc(-n3cc(C4CC4)nn3)cn12 S(=O)(=O)(c1cc(Cl)c(F)cc1F)N1CC(C)OC(C(F)(F)F)C1(C)C N1(C(c2c(C)oc(CO)c2)=O)CC2CCCC2(CNC(=O)CCC=CC(C)C)C1 CCCC(O)C(=O)N1CC(C(=O)NC2CCOC2C)(COC)C1 c1(C(=O)NCC2N(C(c3c(C)cn(C)n3)=O)CCC2)cc(O)ccc1N c1(CC(=O)NCc2csc(-c3ccoc3)n2)ccc2c(c1)OCCO2 c1(CC)cc(C(=O)NCCC2CN(C(C3CC34CCOC4)=O)C2)nn1C C1(=O)N=C2C=CN(N2)C(=O)NC12CC2.c1(C(C)=O)[nH]nnc1C CN(C)S(=O)(=O)N(C)CC(N1CCN(C(C2CC3CC3C2)=O)CC1C1CC1)=O N1(C(C(C)SCC)=O)CCN(C)C(CNC(=O)C=Cc2cc(OC)ns2)C1 C(N=c1[nH]cnc(C)c1OC)NC1CN(C(c2[nH]cc(OC)c(=O)c2)=O)C1 C(CC(O)CC(=O)NC12CC1CN(C(c1oc(C(F)F)cc1C)=O)C2)SC c1(C(N(CCC(F)(F)F)C)=O)ncn2c1CCC2 N1(C(C(=O)NC(C)C)=O)CC(C)(C)OCC1CNC(c1ccc(F)c(F)c1F)=O N1(C(COC(C)(C)C)=O)CCN2CCN(C(c3ncco3)=O)CC2C1 N1(C(c2c(CNC(C(CCC)OC)=O)noc2)=O)CCOC(C)C1CO c1(C(C(=O)NC2CN(C(CCOCC)=O)C2)C)ccc(F)cc1F n1(CC)ncc(C(=O)Nc2cccc(NC(=O)C(C)(C3CC3)OC)c2)c1C1CC1 c1cc(C2OCCO2)c2c(c1)CCN(N1CCOCC1C1CCC1)C2 c1(NC(N(CCS(C)(=O)=O)CC)=O)ccc(OC(=O)COC(C)(C)C)cc1 N1(C(C(CCC)C)=O)CCN(C(=O)COc2c(C)cccc2Cl)C(CCO)C1 C(=O)(C1CCCn2cncc21)N1CCC(N(C(C(C)n2cccc2)=O)C)CC1 N1(C(c2ncccn2)CC)CC2CC(NC(=O)C(C)OCC3CC3)CC1C2 c1(C(=O)NCC2(CNC(C3CCN(C4CCSC4)CC3)=O)CC2)ccc[n+]([O-])c1 CC(CC(=O)N1CC(C)C1C(=O)NCc1ccc(O)cc1F)C(F)(F)F C1(C(=O)NCC2C(NC(C)=O)CCC2)COCCN1Cc1ccccc1 C#CCCCCCNC(=O)CC1(C)CCN(C(=O)C(C)(C)N(C)C)C1 C12(C(N(C(C)C(=O)NCCCP(C)(C)=O)CCC)=O)CCC(C1)C2(C)C C1(C(N2CCC(C(=O)NCC(C(=O)NC)C)C2)=O)COCC(C)O1 Cc1cccc(C(N2CCCC2CC2CCCCN2C(=O)ON(C)C)=O)c1 N1(C(c2c(OC)csc2)=O)CCN(C(c2cc(CO)n(C)n2)=O)C(C(C)C)C1 c1(CNC(C(C)N(C(C2CC23CCOCC3)=O)C2CC2)=O)cccc(F)c1O C(=O)(C1=CC2CC=CCC12)N1CCN(C2CCN(C(CC(=O)OC)=O)CC2)CC1 C#Cc1ccc(F)cc1C(=O)NCC1CN(C(C2(N(C)C)CCC2)=O)CCCO1 C(=O)(CCC(F)(F)C(F)F)NCC1(NC(C(c2ccc(C)cc2)F)=O)CCC1 C(=O)(CCC(=O)NCC1CCN(C(C2CCS(=O)(=O)C2)=O)CC1)OC C1(C(=O)NCC2OCCN(C(c3cccc(SC)n3)=O)C2)CCCCNC1=O N1(C(C2CC2NCc2ccc(C(F)F)cn2)=O)C2CCC1COC2 C1(C(N2C(c3ncc(C)s3)CCCC2)=O)CC(O)C(N=[N+]=[N-])C1 N1(C(c2nc(COC)oc2)=O)CCC12CN(C(c1cc(Cl)c(C)cn1)=O)C2 C1(C(F)(F)F)(CNC(c2n(C(C)(C)C)nnn2)c2cscc2Cl)CCCCCC1 Cc1cc(Cl)ncc1CC(=O)N(C1CCN(C(C2CSCC(=O)N2)=O)C1)C C(=O)(C(C)C(C)(C)C)NC1(CC(=O)NCC2C(C)COCC2)CCSC1 c1(CCC(=O)NC2C(CNC(C3CN(S(CC)(=O)=O)C3)=O)CC2)ccccc1C c1(CNC(C2CC(O)(CNC(C=C(C)C(C)C)=O)C2)=O)cc(C)cc(F)c1 N1(C(=O)NC(C)CCc2ccc(Br)cc2)CCSCC1(C)C c1(OC)c(C(N2CC(CNC(=O)C(C)(C)CO)C(C)C2)=O)oc2ccccc12 N1(C(C(C(C)OC)NC(=O)CC2CCCN2C)=O)CCN(C)CC(O)C1 C1(CC(=O)N(C2CCN(C(C3(C)CC3(F)F)=O)CC2)CC#C)CCOCC1(C)C c1(CN(CCOC)C(=O)NC(C)CSC)ncnn1-c1ccccc1 N1(C(c2c(CC)ccs2)=O)CCC(C)(CCNC(=O)CC(C)C2CCCC2)CC1 C1(O)(CCC)CCN(C(=O)CCCC(C)NC(c2cnc(O)o2)=O)CC1 C(=O)(C(F)(F)C(O)C1CC1)N(C1CC(NC(c2ncn(CC)c2)=O)C1)C C1(C(=O)Nc2cc(C)sc2)N(C(=O)CCc2ccsc2)CCC1(C)C CCCCC(CC(=O)NC1CCCCCC1O)NC(C1CCC2(CCC2)O1)=O c1(NCC(C)CN(C(=O)C=CCN2CCCC2)C)snc(Cl)c1C#N CC(C(C)(C)C)=CC(=O)NCC(O)CN(C)C(c1cc(C2CC2)sn1)=O C(CC)(C(=O)NCCCCc1cnc[nH]1)N(C(C(C)NC(CC)=O)=O)C c1(C(=O)NCCC(CC)(C)NC(c2ccco2)=O)cc(F)ccc1O CCC(O)C(F)(F)C(=O)N1CC=C(C(=O)NCc2ccc(CO)cc2)CC1 c1(C(N2CC=CC(NC(c3cc(C)c(C)nn3)=O)C2)=O)cc2ccc(F)cc2s1 C1(C(=O)NCC2C(NC(c3cn(C(C)(C)C)nn3)=O)CCC2)CC2(C1)CC2(F)F C1(CNC(C(C=C)(F)F)=O)CC2CCCC2N1C(=O)Cc1cncnc1 C1(NC(c2nc(C)c(C)s2)=O)CC(C(=O)NCC2CCOC2(C)C)C12CCC2 N1(C(C2(C#C)CCC2)=O)CCN(C(c2[nH]ccc2C)=O)C(CC)C1.SC CC#CCC(C(=O)NC1CCCC(C)C1)NC(=O)CC(C)C c1(C(N(C2CCC(NC(c3cnn[nH]3)=O)C2)C)=O)noc2ccc(Cl)cc12 C1(C(N2C(CNC(C(c3ccc(F)cc3)C)=O)CCC2)=O)CCc2nn[nH]c2C1 C1(C(CC)CC)CN(c2cc(N(C)Cc3cccnn3)ncn2)CCO1 n1(CNC(=O)OC(C)(C)C)cnc2ccsc2c1=O.C1(=O)C(CC2OCCO2)O1 c1(CC)[nH]c(=N)sc1C(N1CCC(N(C)C(c2c[nH]nc2C)=O)C1)=O c1(CNC(CN(CC#C)C(c2cnsc2C)=O)=O)cn(C)nn1 C1(C(N2C(CNC(C)=O)CCC2)=O)CCN(C(C2(C)CC2)=O)CC1 C1(NC(C(C)SC(C)C)=O)C2CCCN(C(c3ccns3)=O)C2C1(C)C C(=O)(C(CCC(N)=O)n1cc(-c2cscn2)nn1)NC(c1ncc[nH]1)CC C(C(C)(O)C(=O)NCCC1CCCN(C(C2CC(C)=NO2)=O)C1)OC c1(NC(C2C(O)CCN(Cc3c(C)c(Br)cnc3)C2)=O)cc(C#N)ccc1F c1(C(=O)NC2C(NC(C=CC(CC)C)=O)C2)cccc(OCc2cscn2)c1 N1(C(CNC(=O)OC)=O)CCC(N(C)C(c2ccnc(OC)n2)=O)C(C)C1 C(N=C(NCC(F)F)NC1CC1c1cccc(Cl)c1)c1cnn(C)n1 N1(C(C2CC(C)C2)=O)CCN(C(=O)C=Cc2ccsc2)C(c2ncc[nH]2)C1 C(CC(CNC(c1coc(C2CCOCC2)n1)=O)NC(C1CCCSC1)=O)OC N1(C(C2CC3CC2C3)=O)CCCC(C2CCN(c3ncc4ncnc-4[nH]3)C2)C1 C12(NC(c3c(SC)scc3)=O)CCCCC1N(C(=O)C(F)F)CC2 n1(CC)nnc2c1C(C(=O)Nc1ncccn1)CN(C(C1(C)CC1)=O)C2 C(CC(O)C(=O)NCCN1CCC(NC(=O)CCN(C)CCO)CC1)OC CC(C)CN(Cc1cccs1)N(C)Cc1ccc(C(F)(F)F)c(F)c1 C1(CC)CN(C(c2cnco2)=O)CCN1C(=O)C(COC(C)C)NC(C)=O CCCC(CC)C(=O)NCc1ccc(C(=O)NC2(C)CC(F)C2)nc1 N1(C(C(CC(=O)OCC)C)=O)CCC2(CCC(NC(=O)CN(C)CC)C2)CC1 Cc1cn2ccnc(C(N3CC(NC(=O)C(F)CC4CCCC4)C(F)C3)=O)c2n1 C1(C)(C(N(CCC(c2cccs2)NC(C2CCC(C)O2)=O)C)=O)COC(=O)C1 c1(C(N2CCCC(O)(CCNC(C(C=C=C)C)=O)C2)=O)cccc2sccc12 N1(C(CCCC#N)=O)C2CCC1CN(C(=O)CC13CC(c4ccccc4)(C1)C3)C2 N(C1CCC(=O)c2ccccc21)C(=O)C1=NOC2COCC12 Cc1nc(C(=O)NCCOCCCNC(C2CC(C)(O)C2)=O)c(C)n1C1CC1 C1(NC(C(CNC(c2sccc2C)=O)OC)=O)CC2CCCC(C1)C2 Cc1cc(C(=O)NCc2ccsc2C(=O)NCCCOC2CC2)c(O)nn1 C#Cc1ccc(C(=O)NC2C3CN(C(=O)C(c4ccc(F)cc4)CC)CC23)nc1 c1(CC)cnccc1C#N.C12(C(=O)NCCCC3CCCC3O)CCCN1C2=O c1(C(=O)NC(C2CCCC2)CNC(C(C2CCC2)OCC)=O)cscc1C(N)=O C1(C(=O)NC(C(N2CC(CC)(OC)C2)=O)COC)COCC1(C)C N1(C(C(C=C)C)=O)CCC(N=[N+]=[N-])(C(=O)NC2CC3C=CC2C3)C1 N1(C(C(CCSC)O)=O)CC(=O)N2CCOCC2(CNC(C2CCCN2C)=O)C1 C(C#Cc1ccccc1)N(C)C(C1CN(S(=O)(=O)CC(F)(F)F)CCN1)=O N1(C(C(F)OC)=O)CC(NC(c2ccccc2O)=O)C(C(F)F)C1 C(C)(C)(CCCC(=O)NCCC(C)SC)NC(C1CCC(OC)CC1)=O c1(C(N2CC(NC(C(C)(O)C3CCOCC3)=O)C2)=O)ccccc1F C1(N(C(CCCc2ccc(C)s2)=O)C)CCCN(C(c2c[nH]cc2C(C)C)=O)C1 C1(NC(C2(CNC(C(COC)N(C)C)=O)CC(C)(C)C2)=O)CC2(C1)CC21CCC1 c1(CCC(=O)NCCC(OC)OC)ccccc1[N+](=O)[O-] c1(C(=O)NC(CNC(COc2ccc(OCC)cc2)=O)C)cc(C)ccc1C C1(C(=O)NCCC(C)NC(c2ccc(C(F)(F)F)o2)=O)(CO)CCCO1 C1(C(=O)NCCC2(OC)CN(C(=O)C(C#N)C3CC3)C2)CN(C(C)=O)CCO1 N1(C(C(c2cnccn2)C)=O)CC2CC2(NC(=O)CSCc2cccc(Cl)c2)C1 CC1(C)CC(CNC(c2cccnc2CO)=O)CN1C(=O)Cn1ncccc1=O c1(SCCC(N2CC(CN(C)C(C3CC3(Cl)Cl)=O)C2)=O)ccccc1 c1(C(=O)NC(C)CCNC(C2CC2F)=O)cc(F)cc(S(N)(=O)=O)c1 C1(C(N2CCC2COCc2ccccc2)=O)CCN(C(C2(C3CC3)CC2)=O)CC1 c1(CC)sc(C(N2CCC(C(C)NC(=O)CS(=O)CC)CC2)=O)cc1C N1(C(=O)COCCC2CCCC2)CCCN(C(c2cnn(CCO)c2)=O)CCC1 c1(C(=O)NCC2(NC(c3ncc(Cl)s3)=O)CCOC2)ccc(O)cc1 N1(C(CCCc2c(C)ccs2)=O)CCC2(CCCC2NC(=O)CCC2CCC2)C1 c1(C(=O)NCCC=C=C)ccccc1C(=O)N(CC=C)Cc1ccccc1 N1(C(c2n(C(CC)C)ncc2)=O)CC2CCC1C(CNC(=O)C=CC=C(Cl)Cl)C2 C1(CNC(C=C(COC)C)=O)CN(C(=O)C(=O)NCCC(N)=O)CC12CCC2 c1(C(N2C(C)CC(CNC(CC(=C)Br)=O)C2)=O)ccc(Cl)cc1F C(=O)(C(CC(C)CC)NC(=O)Cc1cnn(CC)c1)NC(CCC)C1CC1 N1(C(c2c(C)nn(CCC)c2C)=O)CCC(Nc2ncncc2Cl)C2(CCC2)C1 N1(C(CSCc2nnc(C)s2)=O)CCCCCC1COC(C1CC2CC2C1)=O c1(NC(C(CCC)F)=O)ccc(=O)n(C2(COCC)CC2)c1 N(C(=NCC(C)C)NC(C1CC(=O)N(C)C1=O)c1cccc(Cl)c1)C1(CCC)CC1 c1(C(=O)NCC(C)N(C(C(C)Nc2scc(C)n2)=O)C)ccc(C2CCC2)nc1 Cc1cc(C)c(NC(=O)C(C2CCN(Cc3cc(F)cc(I)c3)CC2)C)cc1C N1(Cc2ccc(C(=O)Nc3cnc(OC)c(Br)c3)cc2)CCC=C(C(=O)OC)C1 C12(C(=O)NCC3(COCC)CC3)CC(CO1)N(C(=O)CNc1ncccn1)C2 C(C(=O)Nc1c(C)c[nH]c1CC(N)=O)(C(C)(C)C)n1cc(CN(CC)CC)nn1 c1(OC)ccc(CC(N2CCCC(NC(c3cnc(Cl)[nH]3)=O)C2)=O)cc1Cl C1(NC(c2ncn(C)n2)=O)CC(CNC(=O)COCC2CCCC2)C12CCC2 n1(CC(=O)NCC2C=CCN2C(=O)C=Cc2cccs2)nc(Cl)ccc1=O N1(C(C=C(CC)C)=O)CCC(C2(NC(=O)CN3CCS(=O)CC3)CC2)C1 N1(C(C=NOC)=O)CCN(C(c2ncccc2F)=O)CC1c1ccccc1Cl c1(C(N2CC(Cn3cc(-c4nc(C)sc4)nn3)C2)=O)ccc2ncccc2c1 c1(C(=O)NCCN(C(=O)CCc2cnn(-c3ccccc3)c2)CC)ccncc1 C(CC(O)C(F)(F)F)NC(CCN(C(C(COCC)C)=O)CCO)=O c1(OC)cccc(OC2(CC(=O)OCC3CCCC(=O)O3)CCC2)c1 C(=O)(C1=C(C)CCOC1)NC1C(NC(CCN(C)CC)=O)COCC1 N12CCC(C(OCC)C1)NC(=O)C2c1cc(Cl)nn1C.C(C)OCC.OCC C1(CNC(C=C(C)C2CC2)=O)COCCN(C(C2CCC(N(C)C)CC2)=O)C1 N1(C(C2N=C(C)SC2)=O)CCCC1(C)CNC(c1cnn(CC(C)C)c1)=O N1(C(Cc2n(C)ncc2)=O)CCC2(CC1)CN(C(C1C(F)(F)C13CC3)=O)CCO2 c1(CC)ncnc(CC)c1C(N1CCOC(CCNC(=O)C(O)CC)C1)=O C=CCC(C)(CC)C(=O)N1CCC(NC(=O)CCCC2CCCCC2)C(O)C1 N1(CCC#C)CCC(C(=O)NC2(CCNC(=O)C(C)C3CCC3)CCC2)CC1 C#CCC(CC#C)C(=O)N1CCC(CF)(NC(=O)Cn2nnnc2C(C)C)C1 C1(C(C)C)(C(=O)NCc2cn[nH]c2)CCN(C(=O)CN2CCCC2=O)C1 C(=O)(CC(C)(C)CC(=O)OC)N1CCCCC(CNC(C(CCC)C(C)C)=O)C1 C(C(=O)N(C1CCN(C(c2ccc(C3CC3)s2)=O)CC1)C)(C(C)C)N.C(N)(=O)OC C(=O)(C(F)CCC(C)(C)C)NCC(C)N(C(c1ccc(C)c(O)n1)=O)C N1(C(CC2CC(=C)C2)=O)CC(C2CCCN(C(C3CC3(F)F)=O)C2)C1 c1(OC)ccc2cc(CC(N3CCN(C(C4CC4Cl)=O)CC34CCC4)=O)ccc2c1 c1(C(N2CCC(NC(CCC(=O)NC)=O)CC2C)=O)cnn2c(C)c(C)ccc12 S(=O)(=O)(CCS(=O)(=O)C(F)(F)F)N(C1(SC)CNC1)C C(CCC)(C(=O)N1CC2CC1C2C(=O)NC(C)C(C)(C)CO)=CCC n1(CC(N2CC(CN(C(CC=CC=C)=O)CC)C2)=O)nc(-c2cccs2)oc1=O C1(C(N2CCC(CCNC(C3CSC3)=O)CC2)=O)CSc2ccccc2O1 C1(NC(COC(CC)(C)C)=O)CCCCC1CNC(=O)C(n1ccc(C)n1)C C(C(=O)N1CCCO1)NC(C(C1CC(C#N)C1)NC(C1OC2CCC1C2)=O)=O C1(CC(=O)NCCc2cn(C3CCC(C(=O)O)C3)nn2)Cc2cccc(Cl)c2O1 O=S(=O)(c1ccc2nc(N3CCC(=C(F)F)CC3)sc2c1)NC1CCCC1O c1(C(N(CC(O)CNC(=O)CCn2ccnn2)C)=O)ccc(C2CC2)s1 C12(C(=O)Nc3cc(CC)c(F)cc3)CCN(C(=O)C=CC3CC3)CCC1C2 C(=O)(CC(CCC)NC(c1conc1C)=O)N1CC(=C)C1 C1(C(=O)NCC(CNC(COC)=O)O)CCc2nc(C)cn2C1 CC1CN(C(=O)CCCS(N)(=O)=O)CC(C)N(C(=O)Cn2ncccc2=O)C1 O=C(C(F)CC1CN(C(C2C=CCS2)=O)C1)Nc1cnn(CCF)c1 C(=O)(CCCC(=O)NCC1CN(C(=O)C(C)N2CC(OC)C2)C(C)(C)C1)OCC c1(C(N(C2CCN(C(=O)COC3CC3)C2)CCC)=O)cnn2c(C)cccc12 c1(C(=O)NCC2CC(NC(C3(OC)CCCC3)=O)C2)cnc2occc2c1 C(=O)(CC(C)CC(F)(F)F)N(CC(C)NC(Cc1nnc(C)o1)=O)C c1(CNC(C)(CCBr)c2nnnn2C2CCC2)cccc2ccsc12 C1(C(N(CCN(C(c2n(CC(C)C)ncc2)=O)C(C)C)C)=O)CC2C=CC1CC2 C(C(=O)NCCC1CCN(C(=O)C(F)n2cccn2)CC1)(C(C)(C)C)SC Cc1cnc(N)c(C(N2CC(CNC(=O)CCOC(C)C)CC2(C)C)=O)c1 c1(C(N2CC3C(NC(C4C(CC)OCC4)=O)C3C2)=O)cc(Br)c(=O)n(O)c1 c1(C(=O)NC2CN(C(c3cnc(SC)n3C)=O)CC2F)cccc(Cl)c1C C(C)(C)(CCCC(=O)N(C)CC1CC1)NC(C(COCC)C)=O Cc1cc(C(=O)NC2CCN(C(C3CSC3)=O)CC2F)ccc1-c1ccncc1 c1(C(=O)NCC2(CNC(C3N(CC)CC3)=O)CC2)ccc(CSC)cn1 N1(C(C(C(C)C)O)=O)CCCOC(CNC(=O)CCNC(=O)C=CCl)C1 N1(C(N2C(C)C(NC(C3CCOCC3O)=O)CCC2)=O)CCOc2ccccc21 C1(C(=O)NC2(CNC(CC(C)n3cccc3)=O)CCC2)COC2(CCC2)C1 C(=O)(C(C)(C)C1=CCN(C(=O)C=C2CCC2)C1)NCC1CCN(CCC)C1 c1(C(=O)NCC2C(C)CCCN2C(c2cncc(F)c2)=O)cc([N+](=O)[O-])nn1C O=C(NNc1c(F)ccc(F)c1Cl)c1cc(S(=O)(=O)N2CCOCC2)c[nH]1 C1(NC(CCCCOC)=O)CN(C(=O)CCc2cc(C)no2)C2CCCCC12 c1(C(N2CC(C)N(C(C3CCCC34CCC4)=O)CC2)=O)coc2c1C(O)CCC2 CC(C)C(CCCO)NC(=O)CC1(N(C)C(c2ccc[nH]2)=O)CC1 Cc1ccc2nc(C(=O)NC3CC(C)CN(C(c4cc(C)ns4)=O)C3)cn2c1 C1(NC(CONC(c2sccc2Cl)=O)=O)CCCCCC1CO Fc1ccc(N=c2scc(-c3ccoc3)n2CC2CCC(F)C2)cc1 c1(C(N2CCN(C(Cc3nc(=N)[nH][nH]3)=O)CC(O)C2)=O)coc2c(F)cccc12 C(=O)(CN=c1cc(Cl)nc(C(C)NC)[nH]1)N(CCNc1cnn(C)c1)CC C1(CC)CCC(C(=O)NCCCC(C)NC(=O)COCCN(C)C)CC1 N1(C(C2(C(F)(F)F)CC(=C)C2)=O)CC(NC(=O)C(CC)SC)C(C)C1 N1(C(c2cc(C(C)C)cc(C(F)(F)F)c2)=O)C2CCC1C(O)CCC2O C=CCC(C)(C(=O)N1CC2(CC2)CC1CNC(=O)C(CC)CCOC)N(C)C C1(CC)CN(C(c2sc(O)nc2C)=O)CCN1C(c1cc(Cl)ccn1)=O C(CC(C(=O)NC1(CO)CN(C(=O)CC2(N(C)C)CCCC2)C1)NC=O)SC N1(C(C(CC)OC)=O)CC2CC(NC(c3c(OC)nsc3OC)=O)C(C2)C1 CCC(CC(=O)NC(C)C(CO)NC(C1CC12CC2)=O)CC(C)C c1(C(=O)NC2CCCC(NC(c3ccc(C)nc3)=O)CC2)ccc2occc2n1 C(c1ccc(C(F)F)o1)=CC(=O)N(C)CC1CCN(C(C(C)OCCOC)=O)C1 C1(CNC(c2cc(OC)no2)=O)CCC(CN(C)C(c2ccccc2Cl)=O)CC1 c1(-c2cc(C(=O)NCC3CCN(C)C3)sc2)cccc2c1CCCC2 c1(NCC2C(C)C2C)ccccc1CSc1ccccc1 c1(CN(C(c2nc(C(C)(F)F)no2)C)C)nnc(C2CCOCC2)o1 N1(C(C2C(CC)OCC2)=O)C2CCCC1CN(C(=O)C1=CC3CCC(C1)C3)C2 N1(C(C(C)NC(C)(C)C)=O)CCC2(CCC(CNC(c3ccoc3)=O)CC2)CC1 CCCCC(C(=O)N1CCN(C(c2cc(OC)n[nH]2)=O)CC1)N(C)C c1(C(=O)NCC(CO)NC(c2c(CC)cccn2)=O)ccc2nonc2c1 c1(CC(N2CCCC(NC(C3(C=C)CC3)=O)C2)=O)ccc(C)c([N+](=O)[O-])c1 C(=O)(CCS(C)(=O)=O)NCCC1N(C(c2nccc(SC)n2)=O)CCSC1 c1(C(=O)N)cccc2nc(O)[nH]c12.C(=O)(C(C)N(CC)CC)NC(=O)NCCCCC C(=O)(CC(O)CC(C)(C)C)N1CCC(NC(CCCC#CC)=O)C(C(N)=O)C1 c1(C(=O)NCC2C(C(=O)NC3CN(C)C(CO)C3)CC2)n[nH]c2c1CCC2 c1(CCC=C)ccc(C(=O)NC2(C)CC(NC(C3CCSC(C)C3)=O)C2)cc1 C(=O)(CCCS(N)(=O)=O)N1C(C(CNC(c2c(C)n(CO)nc2)=O)(C)C)CCC1 C1(OC)CC(CNC(c2cnn(C)c2C2CC2)=O)N(C(=O)CCn2ccnn2)C1 c1(C(N(CCC(=O)N(C)CC2CC2C)CC)=O)ccncc1O c1(SCC)ccccc1C(=O)NCC1COCC1NC(C1CCS1(=O)=O)=O Cc1[nH]nc2c(C(=O)OCC(C3CC=CCC3)=O)cccc12 c1(N(C(C(CC)C)=O)CC2CCCCN2)cnc([N+](=O)[O-])n1C C(=O)(CCCCc1ccccc1)NC1(C)CC(NC(C2CC23CC3(F)F)=O)C1 CCC(CC(=O)NCC(O)CNC(=O)COc1ccn(C)n1)C1CCC1 C=CC(C)(O)C(=O)NCC1CCCN1C(=O)CS(=O)CC C(=O)(CCCC(=O)N1CC2(CNC(c3c(C)cccc3F)=O)CC1CO2)NC c1(N2CCC(CC(CNC(=O)OC(C)(C)C)OC)CC2)cc(O)nc(C)n1 n1(CC(N2C(C(=O)NC3(C)CC(C)C3)C(C)C2)=O)ncccc1=O N1(C(c2ncc(CC)s2)C(=O)NCCC2(C)CC2)CCCC(CC(=O)OC)C1 C1(C(=O)NC2(CC=C)CCCC2)CN(C(c2cnn(C)c2C2CC2)=O)CC1OC c1(C(=O)NC(C)CNC(C23CC(CN(C)C)(C2)C3)=O)cc2c(cc1O)CCCC2 c1(CN(C)C(c2c(Cl)cnn2C)=O)ccc(CNC(=O)CC2CCC3CC23)cc1 C(=O)(C(CC)CC(C)C)NC(CC#CC)C(=O)NCc1ccc(C#N)cc1 c1(C(c2n(CCCC)nnn2)NCC2CC23CC3)cc2ccccn2n1 N1(C(CC2CCN(c3cncc(C)n3)C2)=O)CC2CC(O)C(O)CC2C1 C#CC1(C(=O)NCC2(C)CCN(C(=O)C(c3cnccn3)C)C2)CCOCC1 C(CNC(c1cnsn1)=O)(CO)NC(=O)COCC1CCCO1 Cc1cc(Cl)cc(C)c1C(=O)NCC1C(C)CCCN1C(C1CCS(=O)(=O)N1)=O N1(C(CNS(CCOC(C)C)(=O)=O)=O)CCN(C(c2ncn(C)n2)=O)C(C)C1 C(=O)(C(C)C(O)CC(C)C)NC(CC=CC(=O)NC(CCCC=C)C1CC1)(C)C CC1CN(C(=O)CC#N)CCN(C(C2(c3ccccc3Cl)CC2)=O)C1 c1(C(N2C3CC(NC(c4cn(CC)nc4)=O)(C3)C2)=O)c(Cl)c(CC)nn1C c1(C(=O)NC2(CNC(CC3C(C)=NNC3=O)=O)CC2)cnc(=NCCF)[nH]c1 c1(OC)cc(CN2CCC(O)C(C(=O)NCCCS(C)(=O)=O)C2)ccc1I c1(CNC(c2c[nH]c3ncc(Cl)cc23)c2n(C)nnn2)cc(F)c(F)c(Cl)c1F CC(C)(O)C(C(=O)NC1CCCC1C(C)(C)C)NC(=O)C(=O)NCC(F)F c1(CNC(C2CC(NCc3c(C(=O)OC)ccs3)C2)=O)cn(C)nc1C C(CCCCC(=O)NCCc1ccccc1O)NC(=O)C(F)OC(F)(F)F CCCCC(C(=O)NC1CC=CCC1C(=O)NCC(c1cnc[nH]1)C)N(C)C c1(CC(=O)NC2CCC2CNC(=O)Cc2ccc(Cl)s2)csc(Cl)n1 N#Cc1ccc(SCC(=O)NCC2(O)CN(C(C3CC(F)(F)C3(F)F)=O)C2)cc1 c1(C(=O)NCC2N(C(C(C3CCCC3)OC)=O)CC2)ccccc1C1(C#N)CC1 N1(C(C(C)CF)=O)CCC2(CCCC(CNC(=O)CC3(CS(C)(=O)=O)CC3)O2)CC1 C1(C#N)(OC)CC(C(N2CCC(n3cc(C4CCCC(O)C4)nn3)C2)=O)C1 n1(CC)nc(C2CC2)cc1C(=O)NC1CC(N(C(=O)C(C)OCC(C)C)C)C1 C(=O)(C(C)CC(N)=O)NC(CNC(C1(C)ON=C(C)C1)=O)(C)C1CC1 CC(CCN(CC(=O)OCn1cncn1)C)c1cn[nH]c1 c1(C(=O)NC2CC(NC(c3ccc(C)c(C#N)c3)=O)C2)ccc(S(N)(=O)=O)cc1 c1(C(N(CC(C(=O)NC(CC(C)C)(C)C)C)C)=O)cc2ccccc2[nH]1 N1(CCCOC(C)C)CCC(CNC(c2cscc2C(F)F)=O)C1 C1(C(=O)NC2C=CCN(C(=O)CCC3CCCCC3)C2)CC12CCOCC2 c1(C(N2CC(CNC(c3n[nH]cc3F)=O)OCC2)=O)noc2c1COCC2 N1(C(c2cn(CC)nn2)=O)CCC(C)(NC(=O)C(c2c(Cl)cccc2Cl)C)CC1 c1(C(N2CCCC2c2cnn(C)c2)C(=O)NC2C(C)=C2)cnc2cc(C)nn2c1 C12(NC(C=C(C)C)=O)CCN(C(=O)CCc3ccc(F)nc3)CCC1C2 C(C(CCC)C(=O)Nc1ccc(-n2cccc(C(=O)OC)c2=O)nc1)CC#C c1(SC)ccc(CNC(C2(Cl)CC2CNC(=O)CSc2nc[nH]n2)=O)o1 N1(C(C(C)NC(C=C)=O)=O)CC2OCC(C(=O)NC)C2C1 Cc1cnc(C(N2CCN(C(c3nccc(Cl)c3F)=O)CC2C)=O)c(F)c1 N1(C(C(C)OCC)=O)CCC2CCN(C(C3CCc4n[nH]c(C)c4C3)=O)CC2C1 c1(NCCCN(C)C(c2cnn(C3CCOC3)n2)=O)ncn(C)c(=O)c1Br N1(C(c2n(C(CC)CC)nc(C)c2)=O)CCOC2CCN(C(C3CC3F)=O)CC12 C1(C(C)C)CN(C(c2ccccn2)=O)CCN1C(=O)C=Cc1csc(Br)c1 c1(N(C(C)CCNC(c2ccc(Cl)cn2)=O)C)cc(O)nc(O)n1 C1(C(N(CCC#C)CCOC)=O)CCCCCCN1C(c1conc1CC)=O C1(C)(CC=CCNC(C2(CCOCC)CCCC2)=O)CCCCCC1 C1(C(N(CCNC(C(C)(C)NS(C)(=O)=O)=O)C2CC2)=O)CCCC12CCOCC2 N1(C(C(C)Cc2ccco2)=O)CCCC(C2CCN(C(C34CC(F)(C3)C4)=O)C2)C1 c1(C(=O)NCCN(C(C2CC(n3ccnn3)C2)=O)C2CC2)cnccc1Cl c1(COC)ccc(C(=O)NCC(C)N(C)C(c2cncc(C(N)=O)c2)=O)cc1F N1(C(C)C)CCCC(c2nnnn2C2CC2)(NCc2cc(Cl)cc(Cl)c2)C1 N1(C(CC(C)C)=O)CC(NC(c2nn(C)c(C(F)(F)F)c2Cl)=O)CCC1C Cc1ccc(Nc2ccc(C(C)NC(=O)CCc3cnccn3)cc2)cc1C C(C(=O)NC1(C)NC(=O)NC1=O)(C(C)(C)O)NC(c1nc(OC(C)(C)C)oc1)=O c1(N(CCCCCNC(=O)Oc2ccccc2)C)nccc(Cl)c1Cl N1(C(c2ccc(OC)nn2)=O)CC(NC(c2nc(C)nn2C)=O)CC1(C)C c1(C(=O)NCC(C)N(C(=O)CCSCc2ccccn2)C)cncnc1 c1(CNC(c2cn(C)nn2)C(=O)OC)c(N)cccc1F n1(CCCC(=O)NCC2CCCC2NC(C2CC(CC3CC3)C2)=O)ccccc1=O C1(CCNC(c2cccnc2)=O)CN(C(=O)CNC(C2(Cl)CC2(F)F)=O)CCO1 n1(CC)cc(NC(=O)C(CC(F)F)NC(=O)CC2=CCCC2)ccc1=O c1(C(c2cnsc2)(C)NCC(Cl)Cl)nnnn1C1CCC1 C(=O)(C(O)Cc1cn(C)cn1)NC(CNC(C1(C(=O)NC)CC1)=O)C c1(C(N2CC(NC(CN3CC(C)(C)C3)=O)C(F)C2)=O)cnn2cc[nH]c(=O)c12 S(=O)(=O)(c1ccc(NC2CCOC(C(F)F)C2)cc1Cl)N(CCN(C)CCO)C C1(CC(=O)NCCC2CN(C(C)=O)CCO2)(CNC(C)=O)CCCCC1 N1(C(c2ccc(CN=[N+]=[N-])o2)=O)CC(F)(F)CC1CNC(C1CCC=CO1)=O N1(C(=O)NCC(c2cccc(C(F)(F)F)c2)C)CCC(O)C(CO)C1 c1(NC(C23C(CN(C(c4cc(O)cc(F)c4)=O)C2)C3)=O)cccn2ncnc12 c1(C(=O)NCCC2N(C(c3cnc(C)o3)=O)CCOC2)cccc2nnn(C)c12 C(=O)(C(O)CC(C)(C)C)N1CC(CNC(c2c(C)[nH]c(C(F)(F)F)c2)=O)OCCC1 C1(CC(=O)NC(C)CN(C(=O)CSCC(C)C)C)(C(=O)OC)CCCO1 N1(C(CSC)=O)CCC2(NC(c3cncc(C(F)F)c3)=O)CCCCC12 CC(C)(C)C(CC(=O)NC1CCC(NC(=O)C2Cc3ccc(F)cc32)CC1)C(F)F CC(CCCNC(c1ccn(C2CCC2)n1)=O)NC(=O)CSCC(N)=O c1(C(=O)NC(C2(NC(=O)COCCF)CC2)C)ncc(F)cc1F C(CCCCCNC(c1cnn(-c2ccccc2F)c1C)=O)NC(C(C)SC)=O N1(C(C(C2CCC2)OC)=O)CCC2(CCOC2)C(CNC(=O)CN(C)C)C1 C(=O)(C1=CC(C)(C)C1)N1CCCC(CCNC(c2ccc(CC(C)(C)O)s2)=O)C1 c1(OC)ccc2c(C(=O)NC3CC4CN(C(c5cc[nH]n5)=O)CC4C3)cnn2c1 c1(C2N(C(=O)COCC3CC3)CC2)cn(CC2CCSCC2)nn1 CCCCCC(N=c1[nH]c(=NCC2CC2CC)[nH]c2ccc(OC)cc12)C1CC1 c1(C(N(CCN(C(=O)CC2CCC3CC23)C)C)=O)cc(Cl)ccc1NS(C)(=O)=O c1(C(N(CCC(C)NC(c2cncc(-c3cc[nH]n3)c2)=O)C)=O)ccc(=O)oc1 N=c1nc2c(c[nH]1)CC(C(=O)NC1(CNC(c3cc4c([nH]3)CCC4)=O)CC1)CC2 C12(NC(c3csnn3)=O)CCC(F)(F)CC1CN(C(C13CCCC1OCC3)=O)C2 O=[N+]([O-])c1cc(F)c(CNCCCOCC2CCOC2)c(F)c1 Cn1nc(C(N2CC3CC2(CNC(C2CC(O)C2)=O)C3)=O)cc1C#N N=c1[nH]cnc2cc(C(N3C4CCC3C(CNC(=O)COC(F)(F)F)C4)=O)ccc12 C1(NC(C(N(C(c2cn(CCC)nc2)=O)C)C2CC2)=O)CC(C)(C)C1OC Cc1cc(=NC(=O)C2CCCN(C(=O)N3OC4CCC3CC4)C2)[nH]n1C c1(C(C)O)cccc(NC(C2C=CCN2C(c2ccc(CC#N)cc2)=O)=O)c1 C1(NC(c2cc(Br)sn2)=O)CCCN(C(=O)CN(CCO)CCO)C1 C=CC(C(F)(F)F)NC(=O)C(CCC1CCC1)NC(=O)CCCn1ccnc1 CC(=O)CCCC(=O)N1CCN(C(=O)Cc2ccc(C)cc2Cl)C(CC2CC2)C1 c1(C(N(CC(CC)NC(c2ccc(C(N)=O)o2)=O)C)=O)ccc2occc2c1 O=S(=O)(c1ccc(NCC2CCCCO2)cc1Cl)NCCc1ncccn1 N1(C(C(COC)NC(C2CCC(=O)NC2)=O)=O)CC2(COC(=O)C2)C1 S(=O)(=O)(c1ccc(Br)cc1Nn1cccn1)N1CCCC(NC(N(C)C)=O)C1 C(=O)(C1=CCCOCC1)NC1C(CC)CN(C(c2occc2C2CC2)=O)CC1 c1(C(=O)NC2C(C)(C)CN(C(=O)C3=CCS(=O)(=O)C3)CC2)cccc2ncccc12 Cc1nc2ncnn2c(O)c1CCNC(CC(=O)OC(C)(C)C)C(C)C C(=O)(C#CC1CCCCC1)N1CC(C)(CNC(C2CSCC(=O)N2)=O)OCC1 C12C(CCCN1C(c1n[nH]cc1Cl)=O)NC2=O.c1(CC)ccn(C2CCC2)n1 C1(NC(c2c(OCC)cccc2)=O)CC2CC(NC(=O)C=C(C)C(C)(C)C)C2C1 c1(NC(C2C(NC(C3CC(OCC)C3)=O)CC2O)=O)cc(C)c(F)cc1O C(=O)(C1CCOc2ccccc21)N1CC(CC=C)(NC(=O)C(C)CC)C1 C(=O)(C1SCc2cccnc21)NC(C1(CNC(C(C(C)C)(C)C)=O)CC1)C C1(CCNC(c2nnnn2C2CC2)COC(C)(C)C)CCS(=O)(=O)CC1 O=C1CCN(C(C2CC3(CC3)CN2C(=O)CC2CC3CCC2O3)=O)CCN1 CCC(C(=O)NC1CCC(CNC(=O)C(F)(F)c2csc(C)c2)C1)n1cncn1 c1(C(N2CCN(C(c3scc(C)c3)=O)CC2)=O)cc2c(nc1O)CCCC2O N1(C(CCN(S(CC)(=O)=O)C)=O)CC(CN(C(=O)C(C)N(C)C)C)C2(CC2)C1 N1(C(c2ccc(CNC(C3(CCC)CC3)=O)s2)=O)CC2CCCC2C1 C1(C)(NC(NCC(N2CCCCC2)C)=NCCc2ncccn2)CCS(=O)(=O)CC1 CC(C)(C)C(C)(C)C(=O)NCC(O)CCNC(c1ccc2occc2c1)=O c1(C(=O)NC2CCC(C(=O)NCC(=O)NC)CC2)cc(F)cc(I)c1 N1(C(CC2CC(CC)C2)=O)CC(CNC(=O)C(C)Cc2ccncc2)(OCC)C1 N1(C(Cc2cn(C)nc2)=O)C2CCC(C2)C1CNC(c1cc(F)c[nH]1)=O N1(C(CC2CCCC(C)(C)C2)=O)CCC2(CC1)CC2CNC(=O)CSCC(N)=O c1(CC)ccc(O)c(C(N2CCC(CNC(=O)CC(CC)C3CC3)C(O)C2)=O)c1 CC1=C(C(=O)NCCC(C)N(C(=O)COc2cccc(O)c2)C)CCCC1 N1(C(COC2CC(OCC)OC2)=O)CC(O)(Cn2cc(-c3cccs3)nn2)C1.C1CC1 C1(C(=O)NCc2cc(OC)ns2)C2CCC(C2)N1C(=O)CC1CC2(CC2)C1 N1(C(C2CN(C(C)=O)C2)=O)CCCCC1CNC(c1ncnn1C(C)C)=O Cc1cc2cc[nH]c2cc1C(=O)NCC1CCN(Cc2cc(C#N)ccc2Br)C1 C1(F)(CNC(COCC=C)=O)CCN(C(c2sc(C#N)cc2C)=O)CC1 CN1CC(C)(C)CC1C(=O)NC1(C(=O)NCC2(CO)CCCO2)CC(F)C1 C1(C(=O)NC2C=CCN(C(=O)C=CC3CCCC3)C2)Cc2ccccc2S1 N1(C(C(CC=C)CC)=O)CCC2(CCCN2C(c2cc(C)c(C)[nH]2)=O)C1 C=CCCC(C(=O)N1CCC(O)C(C)C1)NC(=O)C(C1CCCCC1)C c1(C(N2C3C(NC(c4coc(CO)c4)=O)C(CC3)C2)=O)ccnc2ccccc12 C1(O)(CNC(C(C)CC2CCC2)=O)CCN(C(C2CCC(O)CN2C)=O)CC1 CC1(C)c2cccn2CCN1C(=O)NC1CCN(c2ccnc(C(F)(F)F)n2)C1 C(CCCC(=O)N1CCCCC1CCO)NC(CCc1cc(C)no1)=O N1(CC)C(=O)CCC1C(=O)N(CCNC(=O)C(O)COCc1ccccc1)CC C(CCC(O)C(=O)NCCOC1CCCC1)NC(c1nn(C)c(CO)c1)=O Cc1cc(C(N2CCC(n3cc(-c4nccn4C)nn3)C(O)C2)=O)ccc1F C(=O)(CC(C)C(C)(C)NC(c1c[nH]c(=S)cn1)=O)NCC(c1nccs1)C C1(C(=O)NC2(C(=O)NC(C)Cc3nncn3C)CC2(C)C)CC(=O)OC1(C)C c1(C(N2C(CNC(CCCOCC)=O)COCC2)=O)coc2cc(F)ccc12 CC1CN(c2nccnc2F)CC1NC(C1CN(C)C1)=O c1(COC)nc2n(n1)CCCC2NC(=O)C(n1cc(C2CC(F)(F)C2)nn1)C c1(C(N2CC(O)(CCNC(c3c(C)cn(C)c3)=O)C2)=O)c[nH]c2cccc(F)c12 C1(NC(c2ncn(C(C)C)n2)=O)CCN(c2ccc(C(F)(F)F)nn2)CC1O c1(OC)ccc(C(=O)NCCC2(NC(C3CCCCC3O)=O)CCC2)c(Cl)n1 c1(C(=O)NCC2CC(C)N(C(C3C4CCCC34)=O)CC2)ccc(F)c(F)c1F C1(O)(C(C)NC(CC2(COC)CCCC2)=O)CCN(C(C2CCSCC2)=O)CC1 C1(C(N(CCC2CC2)CC)=O)(C(C)C)CCCN1C(=O)CC1(C)CCC1 CN1CCN(C2(C(=O)NC3CC(NC(=O)CC4CC5COCC45)C3)CC2)CC1 C1(NC(C2CC(CC(C)(C)C)C2)=O)CCN(C(c2sccc2C(N)=O)=O)CC1O C1(NC(Cc2c(C)cco2)=O)CN(C(c2nc(Br)c(C)s2)=O)CC1C C1(C(N(CCCN(C)C)CCC)=O)CCCCN1C(C1CCCOC1)=O c1(N2CCC(C)(NC(C3OCC3(C)C)=O)C2)ccc([N+](=O)[O-])cc1-n1cnnn1 c1(NC(C(C)OC(c2ncc(-c3ccc(Cl)cc3)s2)=O)=O)cccc2cccnc12 CCCC(C)CC(=O)NC(CCCOC)C(=O)N1CC(CO)C1 S(=O)(=O)(c1cnc(NCC2CCC=CCC2)c(Cl)c1)NC(c1nncn1C)C N1(C(c2c(C)nn(CC)c2C)=O)CC2(COC(COC)C2)C1 c1(C(N(CC(C)CNC(c2nc(C(C)(C)C)no2)=O)C)=O)ccc(C2CC2)cc1 c1(C(=O)NC2C(C)(C)CN(C(C3(Br)CC3)=O)C2)ccc2ncccn12 c1(C(=O)O)ccc(CN(C(C2CCCC2)=O)C2CC2)nc1.C12CCCCN1C2=O C1(NC(C(C)c2cncs2)=O)CCC2(CCN(C(=O)C(C)(C)C3CCOC3)C2)C1 C1(C(N2CCC(N(C)C(c3sccc3C3CC3)=O)C2)=O)CC2C=CC1C2 C1(CC)(NC(=O)C=C(C)C)CCCN(C(C2(c3ccc(F)cc3)CC2)=O)C1 c1(C(=O)NC(C)CNC(C23CC(CF)(CO2)C3)=O)c(Cl)cncc1Cl C(CCCCC(=O)N1C2CCC1(CO)CC2)NC(C1N(C=O)CCC1)=O N1(C(CCCOCC)=O)CCC(C2CCCN(C(c3ccncn3)=O)C2)C1 C(=O)(CCCC(=O)c1ccccc1)NC(C1CN(C(=O)CC2CSC2)CCO1)C Cc1[nH]c(=NCc2ccc3cc[nH]c3c2)sc1C(=O)Nc1ccc2c(n1)CCC2 C(C)(C(=O)N(CCN1C(=O)CC1)CCN(C)CCO)O.C=CCCCCC.CCC C1(NC(c2n(CC)ccc2)=O)CCCCC1NC(=O)C(N1CCC(C)C1)=O c1(C(=O)NCC#CCNC(CC(C)SC)=O)cc2sc(C)cc2[nH]1 N1(C(C2CC(OC)C2)=O)CC2=C(C1)CN(C(C1CCCC1C1CC1)=O)C2 C(=O)(C1=CCCN(Cc2cc(Br)ccc2C)C1)Nc1cccc(CCC)n1 c1(OC)nccc2c(C(=O)NC3CN(C(=O)CS(C)(=O)=O)CC3F)c[nH]c12 c1(C(N2CCC(NC(Cc3c(C)n(C)cn3)=O)CC2)=O)cc2c(cc1O)OCO2 C(C)(CCC(=O)NC(C)(CNC(=O)CCCCN1CCCCC1)C1CC1)OCC Cc1[nH]nc(C(=O)NCC2CCCN(C(=O)CCn3cnnn3)CC2)c1[N+](=O)[O-] C(CC(C)N=c1[nH]c(=NCCc2c(F)cncc2F)c2cccc(F)c2[nH]1)SC C(=O)(CCCCC(F)F)NCCNC(C(c1cn(C)nc1)=O)=O C1(CNC(CC(C)(C)F)=O)CCN(C(=O)C=CC2CCOCC2)CC1(F)F C12(NC(COCCN(C)C)=O)CCC(NC(=O)C(c3cccnc3)O)(CC1)C2 c1(CC)ccc(C(=O)NCC(O)CNC(c2cnn(C)c2C(F)(F)F)=O)cc1N Cc1ccc(N)cc1C(=O)NC1CCCCC1N(C)C(C12CCC(C)(C1)OC2)=O N1(C(Cc2c(C(C)C)con2)=O)CCOCC1CNC(=O)COCC(F)(F)F c1(OC)cncc(C(N2CCC(NC(=O)CCSC3CC3)C(CO)C2)=O)c1C c1(OC)ccc(O)c(C(N2CCCCC(NC(=O)Cc3cnc(C)s3)C2)=O)c1 c1(C(N2CC3C(CNC(C4CC4C(F)F)=O)C3C2)=O)n[nH]c2c1CCC2 C#CC1(C(N2CCC(OCCNC(=O)C(C)c3cc[nH]n3)CC2)=O)CCCC1 N1(C(c2cccc3c[nH]nc23)=O)CCOC2(C1)CN(C(C13CCCC1CC3)=O)C2 c1(C(=O)NC(C)CNC(C23CC(C)(CCO2)C3)=O)cccc(F)c1C#N C(=O)(C(O)CCCNC(C1(C(C)(C)O)CC1)=O)NCCn1c(C)ncc1 N1(C(c2scc(OC)c2)=O)CCC(NC(c2csc(Cl)c2Cl)=O)C(OC)C1 CC(C(=O)NCC1CC2(CC2)CN1C(c1ccc(O)nc1Cl)=O)S(C)(=O)=O CCCCCCC(CC)(CC)C(=O)NC(CNC(=O)CC1CCC(C)(C)C1)CC C(=O)(C(C)(C)S(=O)(=O)C1CC1)NCC(C)(C)NC(=O)CC1OCCO1 CCC(CC)CC(=O)N1CCCC(C2CCCCN2C(=O)C=CC(C)=O)C1 C1(NC(C(n2ncc(C)c2)C)=O)C2CCC1CN(C(c1cnc(N(C)C)o1)=O)C2 C(=O)(CC(C(F)(F)F)NC(c1nnn(CC)c1C)=O)NCCC=CC C#Cc1ccc(C(=O)N(CCN(C(=O)C=CSC)C)C(C)C)cc1F c1(NC(CC2(N(C(=O)CC3CCCOC3)C)CC2)=O)ccccc1F C1(C(=O)NC(CNC(c2ccc(C(C)C)s2)=O)C(C)C)OC2CCC1CC2 C1(C2CCN(C(=O)CC3(C(F)(F)F)CC3)CC2)(NC(CCS(C)(=O)=O)=O)CCC1 C1(CC(=O)NC(C)(C)CCNC(C2CC(O)C2)=O)COCC1(C)C C1(CNC(CCCCC)=O)CCN(C(=O)CCc2ccc(Br)s2)CC1C c1(OC)ccsc1C(=O)NCC(O)C(=O)NCCCOCCO C=CCC(CC)C(=O)NC1(C2CN(C(=O)C(=Cc3cnn(C)c3)C)C2)CC1 CCCCC(C)C(=O)NCC1(CNC(=O)C(=O)NC2CC2)CC12CCC2 N1(C(C(=O)N(C)CCOc2ccccc2)=O)C2CC2C2CC12 C1(CNC(CC=CCC)=O)CC2(CCN(C(=O)CCSC)C2)CO1 CCC(C(=O)N(C(C)C(=O)NC1CCOC(C)(C)C1)C1CC1)C(C)(C)CC C1(C)(CC)CC(NC(=O)Cc2ccc(C)nc2)CN1C(=O)C=Cc1ccc(C)o1 N1(C(C(CN(C)C)NC(CC2C(C)=NNC2=O)=O)=O)CCn2c(C)cnc2C1 CCC(C(=O)OC)C(=O)N1CC2CC1(CNC(C1CN(C3CCOC3)C1)=O)C2 N1(C(C2CC3(CC(NC(c4cncc(C)n4)=O)C3)C2)=O)CCc2cnccc2C1 Cc1nc(C)c(C(N2CCC3CN(C(=O)CNC(C4CCC4)=O)C3C2)=O)c(C)n1 c1(C(C)C)nn2ccccc2c1C(N1CC(O)CC1C(=O)NCc1ccsc1)=O N1(C(c2nncc(CCC)c2)=O)CCC=C(CNC(=O)CCCC(C)C)C1 N1(C(C(CCC)(C)C)=O)CC=C(CCNC(C2CCC23CCCO3)=O)CC1 C=C(C)C1CN(C(=O)C(C)(C2CC2)N(C(=O)CCN=[N+]=[N-])C)CCO1 c1(-c2cnc(OC)s2)nc(C2OCCc3ccccc32)nn1CC(C)CO N1(C(c2c(C)nn(C)c2)=O)CC2CCOCC2(NC(c2cc[nH]c2C2CC2)=O)C1 c1(CC)ncsc1C(=O)NCC(C(C)C)NC(=O)C(c1cncnc1)C c1(C(C)C)ncc(C(N2CCCC2C(C)NC(=O)CNC(=O)NC2CC2)=O)s1 C1(C(=O)NCCC(=C)CNC(c2cncc(Cl)c2C)=O)C2CCCCCC12 CC1CCCN(C(C2CC(CNC(C3CC4CCC4C3)=O)C2)=O)C1 c1(C(N)=O)ccc(C(=O)NCC2CC(CNC(c3cncn3C(F)F)=O)C2)s1 N1(C(=O)C=CC2CCCO2)CC2(CCCN2C(c2cccc3scnc23)=O)C1 c1(CC(=O)NC2(C(N3CCC(CC)C3)=O)CCC2)ccc(F)cc1 c1(CC)ccc(C(=O)N(CC(C)CNC(=O)C(C)N(C)C)C)cc1[N+](=O)[O-] C1(NC(=O)CCOc2ccccc2F)CCCC2CN(C(C3CC(O)C3)=O)CC12 C1(CCOC)(NC(c2ccc(CO)[nH]2)=O)CCN(C(=O)CCC2CCCC2)CC1 C1(NC(C2(C(=O)OCC)CCC2)=O)CCCC1CNC(=O)CCc1cccs1 C1(CNC(c2csc(-c3ccccc3)n2)=O)C2CN(C(=O)CN3CCC3)CC12 N#Cc1cc([N+](=O)[O-])cnc1N1CC2CN(C(=O)CCn3cccn3)CC2C1 C#CCCC(=O)N(C1CCN(C(=O)Cc2ccn(CC)n2)C1)CCO C1(NC(C(OC)OC)=O)C2CC(O)C1N(C(c1cccc3nn[nH]c13)=O)C2 Cc1ccc(C2CC2C(=O)NC(C)(C)C(C)NC(=O)CCc2nncs2)s1 C(=O)(C(C)C(=O)N1CC(F)CC1CN(C)C(C12CSC(C1)C2)=O)OC N1(C(C2(CC=C)CCCC2)=O)CCCC(O)(CNC(c2sccc2COC)=O)C1 C(=O)(CCCC(F)(F)CO)N1CCC(C)(C)C1CNC(=O)CCN1CCCCC1 C1(C(=O)NCc2ccoc2C(=O)NCc2nncs2)CC2(CCC2)C1 CCC(CCC(=O)NC1CC2CC2C1)NC(c1cc[nH]c(=NC)c1)=O c1(OCC)c(Cl)cc(C)nc1C(=O)NCC1(O)CN(C(=O)C=Cc2cccs2)C1 C(=O)(C1=NOC(C)C1)NCC(C1CCCCC1)NC(CC1(CSC)CC1)=O c1(NC2(c3ccc(OC)cc3)CCOCC2)c([N+](=O)[O-])ccc(Cl)c1Cl CC(C)C(C)C(C)CC(=O)N1CCN(C)C(CF)C1 N1(C(C(CN(C)C)O)=O)CCC(CNC(=O)CCc2ccc(F)cc2F)C1(C)C CCCC(CC)(c1nnnn1CCOC)NC1(C)CC1(C)C S(=O)(=O)(c1ccc(Br)cc1Br)NCC1OCCN(C(CCS(C)(=O)=O)=O)C1 N1(C(CN(CCCCCC)C)=O)CCCC(CNC(C2CCC(=O)N2)=O)CC1 C1(C(N(CC(C)NC(c2ccnn2CCF)=O)C)=O)CCC(=O)C1 c1(C(=O)NC2CC(N(C(CC(C)C(F)F)=O)C)C2)ncnc2c1CCCC2 N1(C(CCc2cn(C)nc2)=O)CC(C(F)(F)F)CC1CNC(C1C(C#N)C1(C)C)=O c1(C(N2CC(C#N)C(NC(=O)Cn3cccn3)C2)=O)cccc2[nH]ccc12 C(=O)(C(C)(O)CC(F)(F)F)N1CC(c2ccccc2)(NC(c2c(C)nns2)=O)C1 c1(-c2cn(CCC(N3CC(C(=O)NC)C(=O)CC3)=O)nn2)cccc(O)c1F C(CCS(=O)(=O)c1ccc(NS(=O)(=O)c2sc(Br)cc2OC)cc1)OC c1(OC)ncc(C(N2CCN(C(=O)CSS(C)(=O)=O)C(C)C2)=O)cc1Cl c1(C(C2(C(=O)NCC(C)N(C(CCCCC)=O)C)CC2)=O)cnc(OC)cc1C c1(NC(c2ccncc2)CNC2CCCCO2)cc(N2CCOCC2)ncn1 N1(C(C(F)=CC)=O)CCC(NC(c2ccc(F)c(C(F)(F)F)c2)=O)C(F)C1 Cc1ccc(C(N2CCC(C)C2CNC(C2(n3cccn3)CC2)=O)=O)cc1CO c1(CC(=O)NC2CCN(C(=O)CNc3nccs3)CC2F)ccccc1[N+](=O)[O-] N1(C(C2(C)CCN(C(Cc3cc(C)[nH]n3)=O)C2)=O)CCSCCC1C c1(C(=O)NCC(C)N(C(C(CC)=CC)=O)C)cnc(C(F)(F)F)cn1 CC(C)C(C#N)C(=O)N1CCCC(N(C)C(c2ccc(N(C)C)cn2)=O)CC1 CN=c1[nH]cc(C(=O)NCC2CN(C(C3(O)CC3)=O)CCO2)s1 C(=O)(C(C)(F)C(F)(F)F)NCCC1(O)CN(C(C2(C(C)C)CNC(=O)C2)=O)C1 CC1(C(=O)NCC2CC2CNC(=O)C(c2cccc(N)c2)O)CCNC1=O C(=O)(CS(=O)CCC(F)(F)F)NCCCCCn1cc(CCOC(C)=O)nn1 C(c1ccc(Cl)cc1F)=CC(=O)NCC(CNC(C1CC2CC2C1)=O)OC C1(NC(=O)Cc2ccn(C3CCCC3)n2)CC2CC1N(C(c1n[nH]cc1Cl)=O)C2 CCC(Cc1ccccc1Cl)C(=O)NCCN(C(=O)C(C)NN(CC)CC)C(C)C c1(OC)ncc[nH]c1=NNC(=O)CC(N)C(C)(C)C C#CCC(CC(F)F)NC(C1(F)CN(C(C2CCC(F)C2)=O)C1)=O C1(NC(C2OCCC(C)(C)C2)=O)CCC2(CCN(C(C3(CO)CCOC3)=O)C2)C1 CC1(C2CC2C(=O)NC2CCCCC2C(N2CCCNC(=O)C2)=O)COC1 C(CCN(C)C(c1cc(Cl)cnn1)=O)(C(C)(C)C)NC(COCCOCC#C)=O C1(F)(CNC(C=CCOC)=O)CCCN(C(=O)C(C)(C)Oc2ccccc2)C1 C1(NC(CN(C)CCO)=O)CCC2(CC1)CC2NC(c1ccc(C#N)c(F)c1)=O C1(NC(CS(CC)=O)=O)CC2(CCN(C(c3cc4c(cn3)CCCC4)=O)CC2)C1 N1(C(CC(C)(C)O)=O)CC2(C1)CN(C(=O)CCCC1CCC1)CCO2 C1(NC(CCn2c(C)ncc2)=O)CN(C(=O)CC(C)N(C)C)CC2CC12 c1(CC)cc(C(=O)ON2CC=C(CC(=O)OC(C)(C)C)CC2)ccc1Br Cc1cc(C(=O)Nc2ccc(OC(F)F)c(F)c2)n2nc(C)cc2n1 c1(OCC)cccc(CC(=O)NC2(CCNC(C3CCOC(C)C3)=O)CC2)c1 N1(C(C2C(CCOC)C2)=O)CCN(C(c2cccc3[nH]ccc23)=O)CC(C)(C)C1 CC1(F)CCN(C(=O)C(c2cccnc2)NC(=O)C(F)OC(F)(F)F)CC1 Cc1cccc(CCNC(=NCC2CC2Cl)NCC(C)(C)c2cccs2)c1 c1(C(C)N(C(=O)C(=O)NC2CC2)C)ccccc1F.c1(N)ccccc1 Cc1ccnnc1C(N1CCCC(CCNC(c2ccnc(C(N)=O)c2)=O)C1)=O N1(C(CN(C2CCCC2)C)=O)CCC2CN(C(=O)C3=CCCCC3)C2C1 Cc1ccc(C(C)NC(=O)CONC(c2ccncn2)=O)cc1 N1(C(C2(C)CN(C(C)=O)C2)=O)C2CCC1CN(C(=O)CCCF)CC2 C(CC(C(C)(C)C)NC(c1cc(CO)n(C)n1)=O)N(C(C1CC(C#C)(O)C1)=O)C Cc1cc(C(N2CCCCC2c2ocnc2C(=O)O)=O)cc(F)c1 N(C)(C1=NS(=O)(=O)c2ccccc21)Cc1n(CCC(=O)OCC)nc(C)n1 CCCCCCC(CC)NC(=O)NS(=O)(=O)CC(C)(C)OC c1(C(=O)NCC2(F)CCC(NC(c3c(C)ccs3)=O)C2)cc(O)cc(Cl)c1Cl c1(OCCC(=O)NC2(CF)CCN(C(C(CCC)O)=O)C2)ccc(Cl)c(F)c1 N1(C(C(C)(C)CO)=O)CC(C2(NC(=O)CSc3ccccc3)CC2)C1 n1(CC)ccc(C(N2CC(CF)(NC(=O)C=Cc3cccnc3)C2)=O)c1C N1(C(c2cc(C)oc2C)=O)CC2CCCC2(NC(C2Cc3nnc(C)n3C2)=O)C1 N1(C(c2cccc(C)c2)=O)CC(CNC(=O)C=C2CCN(C)CC2)CC12CCC2 N1(C(C=CCC(C)(C)NC(C2C(OC)(OC)CC2)=O)=O)CCC(C)C(C)C1 C1(Nc2nccc(CC(=O)OC)n2)CCCC12CN(C(c1ocnc1C)=O)C2.CC c12ccc(cc1)S(=O)(=O)N1CC3CCC(C1)C3N2.C(=O)(CC(C)O)SC C(=O)(C1=CCSC1)N(C(C(=O)NC(c1cnn(C)c1)C)(C)C1CC1)C Cc1cnc(C(=O)NCC(C2CCCC2)NC(=O)CN2CCCC2)cc1C#N C1(CCC(C)C)CCCN1C(=O)CSCC1CCN(C(=O)OC(C)(C)C)C1 CC(C)C(F)(F)CC(=O)N1CCCC1CNC(=O)CCC(=O)c1ccc(O)cc1 C(=O)(C1COc2ccccc21)NC1(C)CCN(C(C=C2CCC(C)CC2)=O)C1 C12(C(=O)NCCSCC(C)C)CC(CN(C(=O)CC3CCC(C)O3)C1)C2 c1(C(=O)NC2CCN(C(c3cc(C)sc3)=O)CC2O)cc2sc(C)cc2s1 CN1CCOC(C(N2CC(C(=O)NCCNC(C3(O)CCN(C)C3)=O)C2)=O)C1 N1(C(CCC=C)=O)CC2(NC(c3cnc(C(C)(C)C)nc3)=O)CCC1C2 CN1CCN(C(c2occc2CNC(=O)CC23CCCC2C3)=O)C(CO)C1 C=CCC(CC=C)C(=O)N1CCCC1C(=O)Nc1ccc(F)c(CO)c1 C(CNC(=O)CCc1cnn[nH]1)(CNC(=O)CCOCCN(C)C)OC C1(C(N(CC)CC2CCC2)=O)(CNC(C2COCC2(C)C)=O)CC2(CC2)C1 C1(C(N2CCC(CC(=O)NC(COC)(C)C3CC3)C2)=O)CCCCC1(C)C c1(SCC)ccccc1CC(=O)NC1CCCCC1NC(=O)CC1CC=CCC1 C(=O)(C1=C(Cl)CCOC1)NC1CC(NC(=O)CC(C(F)F)c2ccc(F)cc2)C1 c1(CCCC)cc(C(N2CCCC(NC(=O)CCCNC(C)=O)C2)=O)c(C)o1 N1(C(CCOCC#C)=O)CC(NC(=O)CS(N)(=O)=O)CCC1C C(CNC(C1CC12CCOC2)=O)(CC)(CC)NC(CC1CC(=C)C1)=O C1(C(=O)NCC2(C=C)CCC2)(NC(C2COCC2C(N)=O)=O)CCCCC1 N1(C(=O)CN2CCC2)CCCCC(C2CN(C(c3cnsn3)=O)C2)C1 C(=O)(CCCCN=c1[nH]c(=NC2CC(CC#N)C2)[nH]c2c1CCCC2)NC C1(OCCN2CC(O)(CNC(c3c(CC)cco3)=O)C2)CCC(C)CC1 c1(C(C2N(C(C3CCCN(C(CC(=O)O)=O)C3)=O)CCC2)=O)ccc2c(c1)OCO2 c1(C(=O)NC2CCC(NC(CCCSC)=O)C2)cc2ccc(F)c(F)c2o1 O=C(CCc1cccnc1Cl)NNC(=O)C(=O)c1nn[nH]n1 c12nc(C)c(o1)C(=O)NC2.C1(C)(NC(CC2CC(CC)C2)=O)CCC(C)C1 N1(C(C(CCSC)O)=O)CCC(N(C(=O)CCc2ccsc2)C)C2(CC2)C1 CCCCCC(O)CC(=O)NC1CC(NC(c2ncccc2OC)=O)C1 O=C1CC(C(=O)NC(C(F)(F)F)C2CCCOC2)c2cccnc2N1 N1(C(C(C(C)(C)C)CO)=O)CC2(C1)CN(C(c1coc(S(N)(=O)=O)c1)=O)CCO2 C(CC(C)C)(C(=O)NCCCc1nc[nH]n1)NC(C(CCSC)O)=O N1(C(c2cnc(OC)s2)=O)CCN(C(c2csc(-c3cn[nH]c3)n2)=O)CC(O)C1 c1(C(=O)NC2(c3ccccc3)CN(C(C(N)=O)=O)C2)cnc2c(c1)NCC2 N1(Cc2sc(C)c(I)c2)CCC(C(=O)O)C(C(C)C)C1 N1(c2cc(NCc3nnc(CC)s3)nc(C)n2)CCC(C2CNC(=O)C2)C1 Cc1ccc(Cl)cc1OCC(=O)N(C1CCN(C(c2c(C)nn(C)c2Cl)=O)C1)C C1(NC(C(COCC)n2cc(-c3cc(Br)c(OC)s3)nn2)=O)COCCC1(F)F Cc1cc(F)ccc1C(O)C(=O)NCC1CC1NC(=O)CN(C)C(N)=O c1(C(=O)NCC(CNC(c2cnc(C(C)C)s2)=O)C)cnc2c(c1)CCOC2 CC(Cc1ccco1)C(=O)NCC1(CNC(=O)CCNS(C)(=O)=O)CC1 C=CCC(C(=O)N1CCC(C(=O)NC(CO)CCC=C)C1(C)C)C(C)C C(c1ccc2c(c1)OCO2)=CC(N1CCN(C(C2CCS(=O)CC2)=O)C2CC12)=O C1(C(=O)NC(CN(C(c2ccc(CSCCC)o2)=O)CC)C)CC(C2CC2)C1 c1(C(=O)NCC2(CNC(CCOCCOC)=O)CC2)cc(C)c(C)c(F)c1 N1(C(c2ccc(CC)s2)=O)CCC2CN(C(=O)CC3(CC=C)CCOCC3)C2C1 N1(C(c2[nH]c(=NCC)sc2)=O)CC2CCC1CN2C(=O)C=Cc1ccc(Cl)cc1 C(CC(O)C(=O)N(C)Cc1ccc(CNC(=O)C(O)c2cnc[nH]2)cc1)SC c1(C(=O)O)n[nH]c2cc(C(N3CC4(CCC4)C3c3cccnc3)=O)ccc12 C1(NC(c2cnn(C(F)(F)F)c2)=O)CN(C(=O)C=CC2CCOCC2)CC12CC2 Cc1cc(OCCNC2CC(=O)N(C3CC3)C2c2cccnc2)cc(C)c1 N1(C(CCC)=O)CCC2(CCN(C(=O)Cc3sc(SCCN(C)C)nc3C)C2)C1 C(CCCCC(=O)NC(C(=O)NCC1CCCC1O)C1CC1)=CC Cc1nc(C(N2CCC(O)(CNC(C3CC(C)OC3C)=O)CC2)=O)ccc1C#N CC1CC(c2nnnn2C2CCC2)(NCCCSC(C)(C)C)C1 c1(C(=O)NC(C2CCC2C(=O)NCC(C)(C)n2cccn2)C)coc2ccccc12 C(=O)(CCCCCCNC(C1C(C#N)C1(C)C)=O)NC(C)C(C)(C)O c1(CSC)cncc(C(=O)NC2(C)CCN(C(c3ncccc3C3CC3)=O)C2)c1 C1(CC(N)=O)CN(C(C2(C)CCCN2C(c2ccc(CO)o2)=O)=O)CCO1 CCCCC(F)C(=O)N(CCC(N1CC(CO)(CO)C1)=O)CCO C1(CCNC(CSCCC)=O)C(C)CCCN1C(=O)Cc1nc([N+](=O)[O-])n[nH]1 c1(CC(C)C)cc(C(=O)NCCCNC(C2CC(C)(C)C2)=O)no1 C1(CNC(C(CSC)(C)NC(c2csc(O)n2)=O)=O)CC(C(N)=O)=NO1 CCC(CC(=O)NCC1CC(C)N(C(c2c[nH]c(=O)cn2)=O)C1)CC(C)C C1(C(=O)OC)C2CCC1N(c1nnc(-c3ccc(Cl)cc3C(F)(F)F)o1)C2 CC(CN=c1ccnc(Cl)[nH]1)N(C(=O)CCC1CC1(F)F)C C#Cc1cncc(C(=O)NC2CN(C(=O)Cc3cccn3C)CCC2O)c1 N1(C(C(C=C)O)=O)C2CCC1CN(C(=O)Cc1cccc(OCCC)c1)C2 c1(C(=O)NCCCN(C(c2cnc(NC)cn2)=O)CC)cc(Cl)ccc1Br N1(C(CCOC(C)C)=O)CCC2OCCN(C(=O)C3=NOC(C)C3)C2C1 c1(COC(CCc2c(C)[nH]n(-c3ccccc3)c2=O)=O)cc2cccc(Br)c2s1 C(c1ccccn1)=CC(=O)NCC1C=CC(NC(c2c(C(C)C)ncs2)=O)C1 C1(NC(COC(C)=O)=O)CCN(C(=O)Cc2csnn2)CCC1(F)F C#Cc1cc(C(=O)NCC2CC3CC3N2C(=O)C(CC)N(CC)CC)ccc1C Cc1cc2c(cc1Br)N(C(=O)C(=O)NCCCOC1CCCOC1)CC(C)O2 CCC(CC)C(=O)NCC(C1CCN(C(c2cc(C)n(C)n2)=O)CC1)F Cc1cnc(C(=O)N(CC(C)(C)CNC(c2ccc(C(C)(C)C)cc2)=O)C)nc1 C1(CC)C(NC(=O)C(CO)NC(N)=O)CCN1C(C1(N(C)C)CC1)=O C(C(C(=O)N1CC(CNC(c2cc(OC)no2)=O)C(C)C1)C(C)(C)C)OCC=C C1(C(N2CCC(NC(C3(CC(=O)OCC)CC3)=O)C2)=O)CCC2(CC1)CC(O)C2 Cc1csc2cc(C(=O)NCCC(C)(C)CNC(=O)CC3C=CCC3)[nH]c12 c1(C2C(C(=O)OCC)C23CC3(F)F)ccc(C#N)c(C)n1 C(=O)(C(CCC1CCC1)NC(=O)COC1CCOCC1)NC(C(C)C)C1CC1 CCCC(C(=O)N(C)OCC(F)(F)F)NC(C1CCOCC1(C)C)=O C12(NC(C(CSC)C)=O)CC(C)(C1)OC21CCN(C(=O)CCC[N+](=O)[O-])CC1 N1(C(C2C(CCC)CCC2)=O)CCCC(N(C)Cc2cccnc2C)C1 c1(CC(=O)NCC2CN(C(CCOCC#C)=O)CC2C)c(C)[nH]c2ccccc12 C1(NC(c2n(C)ncc2)=O)CC(CNC(c2n[nH]cc2F)=O)C12CCC2 N1(C(=O)C=Cc2ccc[nH]2)CCCC2(CCN(C(C3CC4C(C3)C4(F)F)=O)C2)C1 CCCC(C(=O)NC1CCCCC1CNC(=O)C=C1CCCCC1)NC(N)=O N1(C(CCOCCOCC)=O)CCC2C(C(=O)NC(C)CF)C2C1 N1(C(c2n(CC)c(O)nc2)=O)CC(C2CC2C(=O)NCC2(C)CC2(F)F)C1 C(=O)(C1=NOC(C(C)(C)C)C1)NCC(CNC(C1(CO)CC1)=O)OC c1(C(N2C3CC(CNC(CC4N(C)CCC4)=O)C2CC3)=O)ncn2ccccc12 Cc1c(C(=O)NCC2(O)CN(Cc3cc(Br)ncc3Br)C2)cccc1I N1(C(CCNC(C)=O)=O)CCCC2(NC(c3cocc3Br)=O)CCCC12 C1(C(=O)NC2C(NC(c3c(-c4cn(C)nc4)c[nH]c3)=O)COC2)CC2C=CC1C2 c1(C(N(CCC)CCNC(c2cnnc(O)c2)=O)=O)cc2c(O)cccc2n1C c1(OC)ccc(NC(=O)CCCCn2cc(C3COCC3O)nn2)cc1Cl C(C(=O)Nc1cccc(I)c1)(C1=CCCCCCC1)N1C(C)CCCCC1 C1(C(=O)NC(CN(C(C2CC(F)CN2C)=O)CC)C)CCCCS1(=O)=O Cc1ncc(C)c(N2CC(CO)(NC(=O)C(C)C3CCC3)C2)n1 c1(NC(C2(NC(C(C)SC(C)C)=O)CC2)=O)cncc(Cl)c1 N1(C(c2c(C)coc2)=O)CCC(C2(NC(C3CCCC3O)=O)CC2)C1 C(=O)(C1=CC2C=CC1C2)NCC(CC)(C)NC(C1CC2CCCCN2C1)=O C1(C(=O)NC(CC)C(C)CN(C)C)CCc2ncn(C)c2C1 N#Cc1ccc(N2CC3C(NC(C4CCC(F)CC4)=O)C3C2)nc1 Cc1nc(O)c2c(n1)CCN(C(C1C=CCN1C(c1cc(Br)ccc1C)=O)=O)C2 c1(OC)cc(C(=O)NCC2CCN(C(=O)CC3CC(SC)C3)C2)ncn1 C1(C(=O)NCCC(C=C)C)COCCN(C(C2(C)CCN(C)C2)=O)C1 N1(C(C(C)N(CC)CC)=O)CCC(NC(=O)C(O)CN(C)C)C1C(C)C C1(CCNC(c2ccc(CCC)[nH]2)=O)C(C)CCCN1C(=O)CC1CC1 C(=O)(C1=NNC(=O)C1)N1C(CCC(=O)NC(C2CCC2)C)CCC1 CCC(CC(=O)NCC#CCNC(c1ccc(OC)cc1)=O)c1ccc(C)cc1 c1(C(N2CCC(CN(C(c3cc(C)[nH]n3)=O)C)C2)=O)ncnc2c1CCC2 C1(CNC(c2c[nH]ccc2=O)=O)CN(C(c2csc(-c3ccco3)n2)=O)CCO1 Nc1c(C(=O)NC2(CNC(c3cccc(Br)c3)=O)CC2)cc(F)cc1F c1(C(=O)NCCOCC)nc(CNC(c2cc(CC)[nH]n2)=O)oc1C C1(NC(CCn2c(C)ncc2)=O)CN(C(C2CCCC3(CC3)C2)=O)CC2(CC2)C1 c1(C(=O)NCCN(CC(C)O)C(C2(C)CC2(F)F)=O)ccccn1 CC1(C)CCC(CNC(=O)CC2CC(F)C2)N(C(=O)CCn2cnccc2=O)C1 CC1(c2nc(-c3ncccc3Cl)no2)Cc2ccc(Br)cc2C(=O)O1 N1(C(CCSC)=O)CC(F)CC1CNC(c1cc(C#N)cs1)=O c1(C(=O)NC2CCC(NC(C3(C)CNC(=O)C3)=O)CC2)cncc2cnccc12 c1(C(N2CC(CC)N(C(C3CC(O)CN3C)=O)CC2)=O)ccc(F)c2ccoc12 C1(NC(CC)=O)CN(C(=O)CCCc2ccc(SC)cc2)CCC1CO C(c1cccc(F)c1)=CC(=O)NCCC(C)CCNC(=O)COC(F)(F)F c1(C(N(C(C)CF)C)=O)cc(C(F)(F)F)ncc1I c1(CC(N2CCN(C3CN(C(C(CC)=CC)=O)C3)CC2)=O)ccc(F)c(Cl)c1F C1(NC(C(C)CC2CC2)=O)CN(C(c2cc(Cl)cn2C)=O)CC1c1cnn(C)c1 C1(OC)CCC(C(=O)N(CCCF)C)C1 C#Cc1ccccc1CC(=O)NC1(C2CCCN2C(=O)C(C)SC)CC1 C(=O)(C1CCSc2ccccc21)N1C(CNC(c2c(F)ccc(C)c2)=O)CC1 Cc1nc(O)ccc1C(=O)NCCN(C(=O)C(F)C1CCCC1)C(C)C N1(C(C2(CCNC(CC(=O)NCC#C)=O)CCC2)=O)CCC(C2CCOC2)C1 C(=O)(CCCNC(N)=O)NC1C(NC(C=C(COC)C)=O)CC1 C(=O)(C(c1cccs1)NC(=O)CSCC(F)F)N(C)CC1CCOC1 C1(CC(N2CCC(C(C)NC(c3cn(C4CC4)nn3)=O)C2)=O)CCCC(C)(C)C1 c1(C(=O)NC2CCCC(NC(c3c(C)n(C)cn3)=O)C2)ccc(C(F)F)c(F)c1 N1(C(C2C(C)C2)=O)CC2CC(C1)CN(Cc1cccc(C3CC3)n1)C2 C(=O)(C(C)(C)C(O)C(C)C)N1C2CN(C(c3cc(CC(C)C)on3)=O)CC1CC2 c1(C(=O)NC2CCN(C(C(CC)Oc3ccccc3F)=O)C2)cc(Cl)cnc1O c1(C(=O)NC2CC(N(C(c3nc(OCC)oc3)=O)C)C2)nn(C)cc1COC c1(C(=O)OC)ccc(S(=O)(=O)N2CCC3(CN(Cc4cnn(C)c4C)C3)C2)n1C C(=O)(CCCCC(N)=O)NC(C(=O)NCC1CC(CC)C1)CO N1(C(C(C)OCC)=O)CCCC(C(=O)N(C)CCONCC(C)C#N)CC1 CC1(C)CCC(CC(N2CCC2C(N2CCCC(N3CCC3)C2)=O)=O)O1 C1(CNC(Cc2c(C)nc(C)s2)=O)C(O)C(O)CN1C(=O)CCc1ccn(C)n1 C1(C(=O)NC2CCC(NC(c3cc[nH]c3C3CCC3)=O)C2)(COC)CCOC1 C1(C(N2CC(OC)C(CNC(COCCOCC)=O)C2)=O)CCn2nnnc2C1 Cc1cc2c(S(=O)(=O)Nc3ccc(OCC#N)cc3)cccc2cn1 C#Cc1cn(C)nc1C(=O)NC(CC(F)F)C(=O)NC1CCCC1OC C1(CNC(CC(=O)OCC)COC)C2CCC(C2)C1N Cc1csc2cc(C(N3CCN(C(C4(C)COCCO4)=O)CCC3C)=O)[nH]c12 c1(C(=O)NC(CCNC(CC(CCC)C)=O)C)cc2cnn(C(C)C)c2nc1C c1(OC)ccc(Cn2cc(-c3nccc(C)n3)nn2)cc1OCC1CCCO1 Cc1c(C(=O)NCC(O)CNC(=O)Cc2ccc(F)cn2)sc2cccc(F)c12 CCC(CC(=O)NC1CCC(O)CN(C(c2nc(OC)c(C)s2)=O)C1)C(C)(C)C C(=O)(C(C)(C)C(C)(F)F)NC(C(=O)NCc1c(CC)nn[nH]1)CC1CCCO1 N1(C(C2C3CN(C(Cc4c(C)n(C)cn4)=O)CC32)=O)C(C)CCC1(C)C N1(C(C2(C(C)(C)C)CCCC2)=O)CCC(NC(c2cc(CO)ccn2)=O)C(O)C1 c1(C(N2CCC(NC(CCOCC#C)=O)C2)=O)cc(C)ccc1NC(C)(C)C N1(C(C(C)OC2CCCC2)=O)CC2(C1)CN(C(c1cccc(=S)n1O)=O)CCO2 N1(C(CCN(C(C(OC)OC)=O)CCO)=O)CC(CO)(CF)C1 C1(C(N2CCC(NC(C3CC4(C3)CC(O)C4)=O)C2)=O)CC12CC(F)(F)C2 c1(CNC(C2C(C)OCCO2)=O)ccc2c(c1)CN(C(=O)CCCC#N)C2 c1(C(=O)NC(C)CNC(=O)C=CC2CCCCC2)cc2sc(Br)cc2[nH]1 c1(N(C(C(C=C)O)=O)C2CCNCC2)ncnc2cccc(OC)c12 c1(C(=O)NC23C(CN(C(c4c(C)cncc4)=O)C2)C3)n[nH]c2c1CC(C)CC2 c1(C(=O)NCCCC2OCCN(C(C3(C)CC3)=O)C2)n[nH]c2c1CCCC2 C12(C(=O)NCC(C)(C)CNC(=O)CC3CCNC3=O)CCC(CC1)C2(C)C O=S(=O)(c1ccc(NCC(F)(F)F)nc1)NCCCNC1C=CCCC1 C#CCC(C)(C)C(=O)NCC1CC1NC(=O)Cc1cc(Cl)n(C)n1 C1(C(=O)NCC(CNC(c2cc(C)c(=O)n(C)c2)=O)C)CCc2n[nH]cc2C1C C1(CC(=O)NCC(COCC)C)CN(C(c2ccn(C)c2CC)=O)CCO1 C(=O)(C1=CC2C=CC(C1)C2)N1CC(CNC(=O)Cc2cccnc2)OCCC1 C=C(Br)CN=c1nc(N2CCc3nncn3CC2)c2c([nH]1)CCC2 C(N=c1[nH]c2c(c(=NCc3n[nH]c(=N)o3)[nH]1)COCC2)c1c(COC)ocn1 C1(NC(=O)C=C2CCSCC2)CCN(C(=O)C=CC2CCOCC2)CC1F N1(C(CCCc2ccc(C)s2)=O)CC(NC(=O)CCNS(C)(=O)=O)CCC(O)C1 N1(C(C2CN(CC)C(=O)C2)=O)CCCC(C)(NC(C2CCOCC2)=O)C1 N1(C(Cc2c(C)nc[nH]2)=O)CC(C)CCC1CNC(=O)CCc1ccc(Cl)cc1 CC(C)(O)C#CC(=O)NC(CC1CC1)C(=O)NC1CC2CC2C1 C(c1ccc(OCC(N2CC=CC2CNC(=O)C(C)N(C)C)=O)c(OC)c1)=CC C(=O)(CCS(=O)(=O)C1CCCC1)N1CCCCC(CNC(C(C)(C)C)=O)C1 CC(C)CC(C(=O)N(CC(C)NC(C12CCC(CO)(CC1)C2)=O)C)C(N)=O Cc1[nH]c(C(C)(C)C)cc1C(=O)NCC1CCCN(C(=O)CC2(O)CCOC2)C1 N1(C(c2cccc(CCC)c2)=O)CC2CC1CN2C(c1cn(C)ccc1=O)=O C12(CN)CCC(N=C3NC(C(F)F)=Nc4ccccc4S3)(CC1)CO2 C1(C(C)NC(C2CSCN2C(=O)C(C)(C)C)=O)CN(C(C2CC=CC2)=O)CCO1 c1(C(=O)NCCC2CC(NC(C=COCC)=O)C2)cc(OC)cc(C)c1N C(=O)(CC(C)(C)C(=O)NCC(C)(CNC(C1CC(C)(C)CO1)=O)OC)OCC c1(CCC)nc(C)c(C(N2CCOC(CNC(=O)CCn3cncn3)C2)=O)s1 N1(c2nnc(C(N)=O)s2)C2CCC1CC(NC(=O)C(C1CCOCC1)F)C2 CCCCCC(=O)NC(c1ccc(CNC(C2CCCN2C=O)=O)cc1)C c1(CC(=O)NCCOCCNC(c2cncc(NC)c2)=O)c(F)cccc1F N1(C(C(C(C)C)n2cccc2)=O)CCC2(CCN(C(=O)C(F)(F)C(F)F)CC2)C1 N1(CC#C)CCN(C(=O)CC(C)CNC(=O)C(C2CCOCC2)C)CC1=O C1(CC(=O)NCC(N2CCN(C(C3(C)CC(C)C3)=O)CC2)C)CCCC(C)(C)C1 CC1CCn2cc(CNC(=O)NCC34CCC(CF)(C3)OC4)nc2C1 c1(C(N(C)CC2CCCN2C(=O)C(F)C2CCOC2)=O)cccc2c1CNC2=O N1(C(C23N(C(=O)Cn4cccc4)CC(C)(C2)C3)=O)CCCC(C2CC2)CC1 c12ccc(nc1)NC2c1nnnn1CCNc1cccc(OC)c1.C1(OC)CC1.CC c1(NC(c2n(CC(=C)C)nnn2)C2(CC)CCCC2)ccc(C2CC2)cc1 C(CC(C)C(=O)N(C)CC1CCCN1c1ccnc(C)n1)OC c1(CC(=O)NC2C(SC)CN(C(=O)Cc3ccon3)C2)c(C)ncnc1C c1(C(N2CC3(C(NC(C4CC45CC5)=O)CCC3)C2)=O)ccc2nc(S)oc2c1 C1(C)(NC(C2CCN(C(CC)=O)C2)=O)CCN(C(c2cc(OC)cs2)=O)C1 C(CCC1CCC1)(C(=O)N1CC(c2ccncc2)C1)NC(C1CC12CC2)=O C1(CNC(=O)CCN(CCO)C(C2C=CCC2)=O)CCCCS1 CC(C)(O)C(F)C(=O)NC1(C2CCCCN2C(=O)Cc2cccnc2F)CC1 N1(CCNC(=O)NCc2ncc(CO)o2)CCC(n2nnnc2C(F)(F)F)CC1 C1(CNC(C2C(CCC)CCC2)=O)(NC(=O)Cc2cnoc2)CC(F)(F)C1 C1(NC(c2conc2C2CCCC2)=O)CCC12CCC2 C1(C(=O)NCCN(CCC)C(C2CCCC(=O)O2)=O)CN(CP(C)(C)=O)C1 C(=O)(C(CC(C)C)OC)N1CC(C(=O)NC(C#C)C(C)(C)C)OCC1 C(=O)(C(C)(C)CS(C)(=O)=O)NC1CCC(NC(C(CCC)CC)=O)C1 c1(C(=O)NC2C(NC(c3cc(C(F)F)[nH]n3)=O)CC2)cc(C(F)(F)F)ccc1F C1(C(=O)NCCOC(C)C)CC2CC2N1Cc1ccc(Br)s1 c1(SC)ccc(CC(=O)NC2CCCC2CNC(=O)CN2CCSCC2)cc1 N1(CCC)CCCC1C(=O)NCCCC1(CNC(C2COC(=O)O2)=O)CCCC1 CC(C)C(CCC(=O)NCC(C)(C)CC(C)O)NC(c1ccsc1Cl)=O CC1(C)CN(C(c2nccnc2C(N)=O)=O)CCC1NC(=O)CN1CC=CC1 C1(NC(CC=CC)=O)CCC(C)N(C(c2cccc(N(C)C)n2)=O)C1 N1(C(CC(C)OC)=O)CC(NC(=O)CCSc2nnnn2C)C(CO)C1 CCC(C)C(O)C(C)C(=O)NC1CCCCN(C(=O)C(c2ccc(C)o2)C)C1 N1(CC(N2CC(CC(N)=O)(NC(=O)COC(F)F)C2)=O)CCC(C(N)=O)CC1 C=CC1(c2cn(CC3CCN3C(C3CCC(=O)NC3=O)=O)nn2)CCOCC1 C1(NC(CCSCCCC)=O)CCCN(C(c2sccc2C#N)=O)C1 c1(C(N(CC(=O)NC2(CCO)CCCC2)C)=O)cn(C)nc1C(F)F N1(C(C(C)c2ccsc2)=O)CC2N(C(C3C=CCC3)=O)CCC2(C)C1 c12ccc3[nH]cc(c3c1)NC(=O)c1ocnc1-2.CC1(C(=O)NCCCl)CCOCC1 c1(C(=O)NC2C(CNC(c3cc(C)c(C)nc3)=O)C2)ccnc2ccc(F)cc12 O=C(C1NCCn2nccc21)NC1CC(N2CCCC2)C1 Cc1cc(NCC2CCN(C(c3cc(C4CC4)on3)=O)C2)c(C#N)cc1[N+](=O)[O-] C1(OC)CN(C(c2ncc[nH]c2=O)=O)CC1NC(c1c(Cl)nsc1Cl)=O CCS(=O)(=O)CC(=O)N(CCC(=O)NCC(C)(C)C(C)O)C C(C(=O)N=c1ccn(CCO)[nH]1)(c1ccco1)NC(C(CCCC#C)C)=O C1(NC(CNC(CCC)=O)=O)CC2CC(C1)N(C(c1nnn(C)n1)=O)C2 CC(C)CC(Cc1ccccc1)C(=O)N1CCN(C(c2ccc(CO)s2)=O)CC1 Cc1nc(CN2CCC(CNC(=O)CC(F)(F)F)CC2)c(C)n1C Cc1cnc(C(N2CC(N3CCCC3)C(C)C2)C(=O)NCCCN(C)C)cc1Br C1(C(=O)NCC2(C)CCOCC2)CCN(Cc2cnc(Cl)s2)CC1O N1(C(c2n(CC=C)ccn2)=O)CCCN(C(=O)CC(C)(O)C=C)CC1C c1(CNC(C2(C(F)(F)F)CCC(NC(=O)OC(C)(C)C)C2)=O)cc(Cl)cnc1C C(=O)(CCN=c1[nH]ccs1)N1CC(C(=O)OC(C)(C)C)(COC)OCC1 N1(C(C(C)OCCOCC)=O)CCC2(CCCC2CNC(=O)CC2CCC2)CC1 N1(C(C(CC)COC)=O)C2CCC1C(NC(=O)Cc1cc(F)ccc1Cl)C2 c1(C(=O)NC(CNC(C(CC)(C)COC)=O)(C)C(C)C)cc2ccncc2[nH]1 C1(NC(c2c(C)ccs2)=O)COCCC1NC(=O)C(C)Cc1ccncc1 Cc1cc(F)c(C(N2CCN(S(=O)(=O)C(C)C)CC2)=O)cc1-c1ccc(F)cn1 N1(C(C(COC)N(C)C)=O)CCCC(CO)(NC(C2CC(NS(C)(=O)=O)C2)=O)C1 c1(CC)ccc(C(=O)NC2CC(C)(NC(c3nc(CC)ncc3Cl)=O)C2)cc1N C1(CNC(c2ccc(CO)cc2)=O)CN(C(OC(F)(F)F)=O)CC(C(F)(F)F)O1 Cc1cc(CNC(C2CCCC2NC(c2cnc(N(C)C)s2)=O)=O)nnc1C Cc1csc(=NCC(=O)N2CCCC(CNC(c3ccc(Cl)cc3F)=O)CC2)[nH]1 CC(C)C(C#N)C(=O)NC1CCCC(C(=O)NCCC(C)(C)N(C)C)CC1 c1(C(=O)NCCC2CC(NC(C3C(C)(CC)C3)=O)C2)scnc1C n1(CC)nc(C)c(C(=O)NC2CC(O)(CNC(=O)C(=O)NC(C)C)C2)c1Cl c1(C(N2CC(C(C)NC(c3ccoc3C3CC3)=O)C2)=O)cn(C)c2ccccc12 CCCCC(C(=O)NCCC1CCOC(C)C1)NC(=O)CNC(C1CC1C)=O c1(C(N(CC(Cc2ccccc2)NC(C(C)CF)=O)C)=O)ccc(S(N)(=O)=O)s1 N1(C(COC2(C)CN(C(C)=O)C2)=O)C(C)CCC1C n1(CC(=O)NC2CCCN(C(CC3CC(C)C3)=O)C2C)nc2ccccn2c1=O Cc1cc(C(=O)N(CCCNC(C2(C(F)F)CCCC2)=O)C2CC2)nn1C C=CCC(CC(=O)NCC1C(CO)C1(F)F)NC(=O)CC1C=CCC1 c1(C(=O)NCC(CC)N(C)C(c2cn(C)cn2)=O)cccc2cnn(C)c12 C(CN=c1cc(C(F)F)nc[nH]1)NC(c1c(Cl)cncc1Cl)=O c1(C(N2CCC(CN(C(=O)CCC(F)(F)F)C)C2)=O)ccc(F)c(F)c1F N1(C(c2ccc(C)cc2)=O)CCN(C(=O)CC2CC(C3CC3)=NO2)C(CCO)C1 C1(NC(CSC(C)C)=O)CN(C(=O)Cc2cc[nH]c2)C2CCCC12 c1(CNC(C2CCN(CC(C(C)(C)C)O)CC2)=O)cccc(F)c1F c1(C(N2CC(NC(C(c3ccccc3)N(C)C)=O)C2)=O)ccnn1CC(F)F CC(C(C(=O)NCC1CCOC1)N(C)CCF)C1CCCOC1 n1(CC(=O)NCC2C=CCN2C(C2CCC2)=O)c(S)nc2ccccc2c1=O c1(OC)cc(C(N2CCC(C(C)CNC(=O)CC(C)C(C)C)CC2)=O)ccc1Cl c1(C(=O)NC2CCCC(N(C(c3c(CC)con3)=O)C)C2)csc2nnsc12 Cc1ccc(F)cc1C(N1C(CNC(=O)Cc2ccccc2F)CC2CC12)=O c1(CC(N2CCC(NC(C(C)(C)SC)=O)C(F)C2)=O)ccc2c(c1)COCC2 c1(C(C(=O)NC2(COC)CN(C(=O)CCC(C)(C)C)C2)C)cccc(C#N)c1 C(=O)(CC(C)(C)CC(C)=O)N1C(CCNC(C=C(C)C2CC2)=O)CSCC1 c1(C(N(CC(C)CNC(=O)Cc2cnnn2C)C)=O)cccc(C#CCO)c1 N1(C(C(CCSC)O)=O)CCCC(NC(c2ccc(N)cc2Cl)=O)CC1 C(CCS(=O)(=O)c1cccc(C)c1)N(C(C(COC)C)=O)C C1(C(=O)NC2(CCCC)CC2)CC2CCN(C(C3CCC=CO3)=O)CC12 N#Cc1c[nH]c(C(N2CC(CC(N3CC3CO)=O)C2)=O)c1 N1(C(Cc2c(C)scc2)=O)CCC(C)C(NC(c2c[nH]nc2-c2ccoc2)=O)C1 C1(NC(C2(C#C)CC2)=O)CCC(C)N(C(c2scnc2CC)=O)C1 N1(C(C)=O)CSCC1C(=O)NC1(C2CCCN2C(=O)CCc2ccsc2)CC1 c1(NC(C2CCCC(NCc3cc(OC)ncc3)C2)=O)cnc(Cl)cc1OC CC1CCN(C(=O)CSc2ccc(F)c(F)c2)CCC1(F)F C(C(C(=O)NCCN(C(=O)CC1COCC(C)O1)C)C(F)(F)F)OC C1(C(=O)NC(CC)CCOC)(CC)CCN(C(=O)Cc2cc(C)on2)C1 C1(NC(C(CCSC)NC(N)=O)=O)CCN(C(C2CN(C)C(=O)N2)=O)C(C)C1 c1(OC)ccc2c(c1)C1(CC1)CN(S(=O)(=O)c1ccc([N+](=O)[O-])c(Br)c1)C2 C1(C(=O)NC(c2c(C)nn(C)c2)C)CCN(C(=O)CCC(C)C)C(C)(C)C1 C1(C(=O)NC(C)(C(=O)NC2CCCCCC2CO)C2CCC2)CC2(CCOC2)C1 Cc1cnncc1C(N1CCCCC1C(C)NC(=O)COCc1ccnn1C)=O C1(CCC)CN(C(=O)C(C)CC#N)CC1NC(=O)CC1CC(C)=NO1 c1(NC(CCOC)=O)ccnc(-n2cc(CC3CCCN(C)C3)nn2)c1 c1(C(=O)NCCC2CCN(C(c3c(C)onc3)=O)CC2)cnc2sccn2c1=O N1(C(C2CCCCC2O)=O)CCC2(C(N3CC(c4ccncc4)C3)=O)CCCC12 C1(C(C)O)COCCN1C(c1ccoc1CNC(=O)CSC(F)(F)F)=O c1(C(N(CCNC(C2CCOC2)=O)CC)=O)cc(S(N)(=O)=O)cc([N+](=O)[O-])c1C N1(C(c2ccc(OC)c(F)c2)=O)C2CCC1CN(C(C1CCOC1C)=O)C2 N1(C(c2ccc(-c3ccc(C)s3)s2)=O)CCC12CN(C(=O)CC1CCCN1C)C2 c1(C2(C(=O)NC3C(OC)CN(C(=O)CC4(C)CCC4)C3)CC2)ccc(C#N)cc1 c1(C(=O)OCC)ccc(C(C)NC(=O)NCC2(c3ccc(F)cc3)CC2)cc1 N1(C(CC(C=C)(C)C)=O)CCC2CN(C(=O)CC(C(C)C)NC(=O)OC)C2C1 Cc1nc(N2CCSCC2CCNC(c2csc(C(C)C)n2)=O)cc(C#N)n1 C1(C(=O)NCCCSCC)CCN(C(=O)c2cccn2C)O1 c1(OCC)oc(C)nc1C(=O)NC(C)CC(C)NC(c1c(C)noc1CC)=O C1(NC(=O)Cn2cc(CN3CCCC3)nn2)CCC(c2ncc[nH]2)CC1 C1(C(=O)OC(C2CCC2n2ccnc2)C2CC2)(COC)CCNC1=O N(C1CN(C(=O)CCSC2CCCC2)Cc2ccccc21)C(C(CC=CC)C)=O C(=O)(C(C)(C)CC(C)C)NCC(CC)NC(=O)C(N1CCCC1)C1CC1 C1(NC(c2ccon2)=O)CCCC12CN(C(c1cccnc1C1CC1)=O)C2 c1(C(=O)NC2(C)CC(NC(c3c(C)onc3)=O)C2)ccc(SC2CC2)cc1 C1(CNC(C(=O)N(CC(c2ccccc2)CC)CC)=O)CCC(=O)N1C N1(C(C(C=C)c2ccccc2)=O)CC2C(CNC(=O)CSS(C)(=O)=O)C2C1 c1(C(C)C)nc(NC(C)(CNC(=O)C2=CC(C)(C)C2)Cn2cccn2)cc(Cl)n1 c1(OC)cc(NC(=O)C(CC(N)=O)NC(c2cnc(O)o2)=O)ccc1C C1(NC(CC2(C=C)CN(C(C3CCSC3)=O)C2)=O)C=CC(C)(C)CC1 Cc1c(C(N2CCC(CN(C(=O)C3=NOC(C)(C)C3)C)C2)=O)cc(O)cc1N C(CCC(F)(F)F)(C(=O)NC1CCC(F)(F)CC1F)Nc1nnc(C(C)(C)C)s1 CCC(C)C(O)C(=O)NCc1cccc(CNC(c2cnc(C(C)C)nc2)=O)c1 Cc1cc(F)c(NC(=O)CC(C(C)C)NC(c2cc(C(C)C)on2)=O)cc1F Cc1c(-c2cnc(NC(c3ccnc(F)c3)=O)s2)cccc1F C1(NC(C(C)OCC)=O)CCCCCC1C(=O)NCC(C)(C)N1CCCC1 C1(C)(C(N2CC(O)(C(C)NC(=O)CC3COC(C)(C)C3)C2)=O)CCC(F)(F)CC1 Cc1nc(C)c(C(C)NC(=O)CCN(C(c2ncccc2C)=O)CC2CC2)[nH]1 C(=O)(C1CCCc2nn[nH]c21)NCC(C)NC(CC(COC)(C)C)=O N1(C(C=CCOCCOC)=O)CC2(CCCN(C(c3cnc(C4CC4)[nH]3)=O)C2)C1 c1(C(=O)NC(C2CCCC2)CNC(C(C)NC(N)=O)=O)ccc(F)c2occc12 C1(NC(CC2CC(C(C)C)OCC2)=O)CCN(CC2CCCCO2)C(C)C1 N1(C(C(C)C#N)=O)CCC(C)(C)C(NC(c2cccc(Br)c2F)=O)C1 C(=O)(C1CCCc2nn[nH]c21)NCC1(C)CC(NC(C2CSCC(=O)N2)=O)C1 n1(CC)ccc(C(=O)NC2CCC2NC(=O)COc2ccc(OC)cc2)c1C CC1CN(C(C2CCCN2C(c2cc(Cl)cc(Cl)c2)=O)=O)c2ccc(F)cc2O1 c1(C(=O)NC2C(NC(=O)CCc3cnn[nH]3)COC2)c(C(F)F)cccc1F C(CC(F)(F)F)SCC(=O)NCC1COC(CNC(=O)CCSCC(N)=O)C1 c1(CNC(=O)NCC2OCCN(C)C2c2ccccc2)noc2c1CCCC2 c1(NC(c2ccc(C(N3CC(C(N)=O)(OC)C3)=O)o2)=O)cc(O)ncn1 C1(NC(CC(c2ccc(F)cc2)C)=O)CCC(Nc2cc(F)ncn2)CC1 n1(C(C)C)nnc2c1CCN(C(C1CC(C3CCNC3)C1)=O)C2 c1(C(=O)NC2CCCC(NC(C=CC)=O)C2)cccc2c(C)[nH]nc12 C(=O)(CCCS(C)(=O)=O)Nc1cnc(Nc2ccc(CC)cc2)nc1 N1(C(c2c(CC)noc2C)=O)CCC(CO)C(NC(=O)Cc2csc(=N)[nH]2)C1 CC1CCN(C(=O)Cc2ccc3c(c2)CC3)CCS1 C1(C)(C(=O)NC2CN(C(C3(C(C)=O)CC3)=O)CC2O)CC2CCC1O2 N1(C(=O)Cc2ccon2)CC2(C(N3CC4C=CC4C3)=O)CC1CCO2 c1(C(N2C(CNC(=O)CC34CCC(CC3)C4)CCCC2)=O)cccc2c1OCC2 CC1(CNC(=O)C=Cc2ccccn2)COCCN(C(c2ccsc2Cl)=O)C1 C1(CC(=O)N(CC(C)NC(=O)C=Cc2cc[nH]n2)C)CC(O)C12CCC2 C1(CCC(=O)NCCNC(C2(CCCC)CCCC2)=O)CCc2cnn(C)c2C1 CC1CCCCC1(CNC(c1cc(F)cnc1O)=O)NC(=O)C=Cc1cocn1 N1(C(CC2(NC(C)=O)CC2)=O)CCCC12CCN(C(c1snnc1C)=O)CC2 C1(NC(C(n2ncc(C)c2)C)=O)CC2(C1)CC(NC(C1(C3CC3)CCCO1)=O)C2 CC1OC(C)C(NC(=O)C(=O)NC2CCS(=O)(=O)C2)C1C CC(C)C(C(=O)NC(C)CCNC(=O)C=Cc1cocn1)n1cnnc1 c1(CNC(CSCC)=O)ccc(CNC(c2cn(C)nc2C(C)(C)C)=O)c(F)c1 Cc1cc(=O)oc(C)c1C(=O)NCCC(C(C)C)NC(c1ccsc1C(F)F)=O C1(COC)(NC(=O)COCC2CCCC2)CCN(C(=O)Cc2n[nH]c(C)n2)C1 c1(C(=O)NC(C2(CNC(c3cccc(=O)n3C)=O)CC2)C)cn2ccccc2n1 C(=O)(C(C(=O)NCC#CCNC(=O)CC(c1ccc(F)cc1)C)OC)OCC C1(CCNC(=O)Cc2ccno2)COCCN1C(=O)Cc1cscn1 c1(C(=O)NC23CC(CNC(c4c(OC)c(Cl)sc4)=O)(C2)C3)cnc2ccnn2c1 c1(C(N2CC(C#N)C(NC(c3ccc(Br)c(Br)c3)=O)C2)=O)cccc2c1CCC2 Cc1cc(O)cc(=O)n1CC(N1CCC(C2(NC(=O)C(C)CN(C)C)CC2)C1)=O c1(C(N2C(C(C)NC(C3C(C)OCC3)=O)CCC2)=O)ccc2c(=N)[nH]cnc2c1 N1(C(C(C)c2ccco2)=O)CCCC(CNC(c2nn(C)nc2Br)=O)CC1 CC(CCC(C)(C)C)C(=O)NCC1CN(c2ncccc2C#N)CCC1(C)C C(CCCC(=O)N(C1CCCC1NC(C1(C(=O)OCC2CC2)CC1)=O)C)SC N1(C(c2sc(Br)nc2Cl)C(=O)NCCOCC)CCN(C)CC12CCCCC2 N1(C(C(C)=C2CCC2)=O)CC(C)C(NC(c2ccc(C)c(C)n2)=O)C(C)C1 C1(NCO)C(CO)CCN1C(=O)CC=Cc1ccccc1.n1(C)ccnn1 CCC(C)C(C(=O)N(C1(C(=O)NCC2CC(N(C)C)C2)CC1)C)OC CC1OCCN(C(=O)CC2CC(O)CN2C(C2CC(=O)C2)=O)C1CO C1(C2CCC2)(C(=O)NCC2C(NC(c3c(C)cc(F)cc3)=O)COC2)CC1(F)F CC1CC(F)(F)CCN1C(=O)C(CNC(c1cccs1)=O)C(C)(C)C N1(C(C(C)OCC=C)=O)CCC(C(C)C(=O)Nc2cccc(O)c2)CC1 C(C(=O)NOCC1(C)CC1)(c1cccc(Cl)c1)OC c1(C(N2CCCC(NC(CC(CCC)C)=O)CC2)=O)c(N)ccc(F)c1F C(CCC)(CC(=O)NCc1nncn1C(C)C)NC(C1(COC)CC(=C)C1)=O C1(N(C(C(C)OCCC=C)=O)C)CC2CCC(C1)N2C(=O)CC1=CCOCC1 C1(OCCCOC)CCN(C(=NCC(C)C#N)NCC2CCCCO2)CC1 Cc1cc(=N)[nH]cc1C(N1CCC(O)(C(C)CNC(c2cnn(C)c2Cl)=O)C1)=O Cc1ccc2c(C(=O)NC3CN(C(=O)CCc4ccn(C)n4)CC3F)n[nH]c2c1 c1(C2(C(N3CC(N(C)C(C4CN(C5CCOC5)C4)=O)C3)=O)CC2)cccc(Cl)c1 C1(CCCC)CCCC1NC(=O)NCC(CO)OCC CC(O)CC(C)CN=c1[nH]c(=NCc2csc(O)n2)[nH]c2c1CCCC2 C1(C(=O)NC2CC(NC(c3ccc(C#N)cn3)=O)C2)C2Cc3c(Cl)cccc3C12 N1(C(CC(=O)NC)=O)CCN(C(C2(COC)CCCCC2)=O)CC1CC(F)F N1(C(c2ncc(OC)cn2)=O)CCN(C(c2cc(OC)ccc2Cl)=O)C2CC12 C1(C(=O)OCC(N2CC(O)CC2C(=O)O)=O)COc2cccc(F)c2O1 C=CC1CCN1C(C1(N(C(=O)C(F)C2CCC2)C)CC1)=O N1(C(C(C)(c2ccccc2)N(C(C)C)C)=O)CCCC(n2cc(CO)nn2)C1 C(=O)(C1=CC2(CCOC2)C1)NC(C1CN(C(=O)CC2(O)CCCCC2)C1)C C(c1ccccc1Cl)=CC(=O)NC(C)CCCCNC(C1CCCN1C=O)=O C(=O)(CCCCCCN=[N+]=[N-])N1CCC(CNC(CC(CCC)O)=O)CC1 c1(C(=O)NC2CCC(N(C(CNS(CC)(=O)=O)=O)C)C2)cccc(C(=O)NC)c1 c1(C(=O)NCC2OCCN(C(CCC)=O)C2)nn(C)c(C(F)(F)F)c1Cl C1(CC)CC(C)CN(C(C2(NC(=O)CC3CCSC3)CCOCC2)=O)C1 C1(NC(CCN(C)CC)=O)C(C)(C)CN(C(=O)C2=NOCC2)CC1(C)C c1(C(=O)NCC(C(C)C)Nc2cc(C(C)=O)ncn2)cc(S(C)(=O)=O)co1 c1(C(=O)NC2CC2NC(C2CC2(Cl)Cl)=O)cc(Cl)ccn1 c1(C(=O)NCC2CCCC(NC(C=CS(C)=O)=O)C2)ccc2nnn(O)c2c1 CCC(C(=O)NCCCCC1CN(C(C2CCC2OC)=O)C1)n1cccn1 c1(C(=O)NCC2(NC(c3c(Cl)cnc(C)n3)=O)CCC2)ccc2c(c1)CC(C)O2 C(=O)(CCC(CF)CF)NC1C(CC)CN(C(=O)CCc2cnc(O)[nH]2)CC1 c1(NC2CN(c3nccnc3)C2)cc(NC2CCCCO2)ncn1 CCCCC(C(=O)NCC1CCC(C)C1)NC(c1cnc(C2CC2)o1)=O c1(C(N(CCCCNC(C(CC)(C)F)=O)C)=O)cnn2c1NCCC2C(F)(F)F c1(SCC(=O)NCC2(OC)CN(C(C3C4CCCCC34)=O)C2)ccc(C)c(C)c1 Cc1cc(C=CC(=O)NCC(O)CNC(C2CC2C(F)F)=O)ccc1OC(C)C C1(C)(NC(c2ncn(C)n2)=O)CCC(NC(c2ccccc2Cl)=O)CC1 c1(C(=O)NCC2N(C(C(CC)COC)=O)CC3(CC3)C2)cn(C)c(=O)n(C)c1=O C1(CCOC)CN(CCNCC2CCCC2)CCO1 c1(C(=O)NC(CNC(C2(CC#C)CCCOC2)=O)C)ccc(C(C)(F)F)nc1C C1(NC(C2(CC#C)CCC2)=O)CC2CCC1N(C(c1c(C)ccc(C)c1C)=O)C2 N1(C(C)=O)CCc2cc(C(=O)N(C3CC(NC(=O)C(C)CO)C3)CCO)ccc21 N#Cc1cc(C(=O)NC2CCCN(C(=O)C(N)=O)CC2F)cc(F)c1F N1(c2cc(C)nc(CO)n2)CCC2CC(NC(c3cc(O)nn3C)=O)CCC2C1 n1(CC)cc(CCNC(C2C(CC3CCC(C(=O)NC)C3)C2)=O)nn1 C1(N(C(=O)CC23CCCC2C3)C)CCN(C(C2(CO)CCOC2)=O)CC1 C(=O)(C(CC)CCCC)NC(CN1CCN(C(CC=CC)=O)CC1)C c1(C(=O)NC(CN(C(c2ccc(OCC)cc2)=O)C)C)cncc(C)c1Cl N1(C(c2c(C)nc(C3CC3)[nH]2)=O)CC2CN(C(C3C4(CC4)C34CC4)=O)CC2(C)C1 c1(CC(=O)NC2CCC(C)(NC(C(C(C)C)F)=O)CC2)ccc2cnccc2c1 CCCS(=O)(=O)C(C)C(=O)NC(C1CCCN1C(=O)Cc1nc([N+](=O)[O-])n[nH]1)C N1(C(=O)Cc2cncnc2O)CC2CCC(C1)N2C(C1CCSC1)=O C(=O)(CC(C)(C)C#N)NCC(CN(C(=O)C(F)C1CCOC1)C)(C)C C(=O)(C(C)(CC)C(=O)N(CC(C)(C)CNC(=O)C=CS(C)=O)C)OC N1(C(C(CC)SC)=O)CCC(O)C1C(=O)NCc1ccn(CC)n1 C1(CNC(=O)C2=CCC2)CCC2(CN(C(c3cc4ncccn4n3)=O)C2)O1 c1(C2(C(=O)NCCC3(NC(C(CCCC)O)=O)CC3)CC2)ccc([N+](=O)[O-])cc1 CC1CCCC1N=c1nc(N2CCC3(CCCN3C)CC2)c2cccc(F)c2[nH]1 CC1CCCCN1CCC(=O)NC1CC(C)(NC(=O)Cc2cn[nH]c2)C1 c1(OC(C)C)ccc(C(=O)NCC2(NC(=O)C=CS(C)=O)CC2)c(O)c1 S(=O)(=O)(c1ccc(N2CC(OC)CC(O)C2)c(F)c1)NCC1(COC)CC1 N#Cc1cncc(CC(=O)NC2CC2NC(c2ccccc2-n2cnnn2)=O)c1 CCC(C)C(O)C(=O)N1CCC(C)(NC(C2CCN(C)CC2)=O)CC1 c1(SC)cc(C(=O)N(C2CC(NC(=O)C(O)Cc3ccccc3)C2)C)ccc1N CC1CN(C(C2(C3CC3)CN(C(=O)C=CC3CCOCC3)C2)=O)CCC1CO c1(CC(=O)NCCN(C(C(COC(C)=O)C)=O)CC2CC2)ccc(Cl)c(C)c1 CC1C(=O)CC1C(=O)NCCCNC(=O)CN(S(C)(=O)=O)C c1(CC(=O)NC(CC)CN(C)C(c2ccon2)=O)ccc2c(c1)CC2 c1(OC)oc(C)nc1C(=O)NCC1CC(NC(C2CCCO2)=O)CC1O C(C1CCCN1C)=CC(=O)NCC1CC(CNC(C2(C(=O)NC)CCC2)=O)C1 C1(NC(c2c(CCC)n[nH]c2)=O)(CO)CCN(C(=O)CC2CC(CC)=NO2)C1 c1(NC(N(CC)CC)=O)cc(F)c2ncccc2c1.N12CC(CC)N(CC1C)C2=O c1(CC)ccccc1CC(=O)NC(C)CC(C)NC(c1coc(OC)n1)=O c1(C(N2CCN(C(CCC(C)SC)=O)CC(CO)C2)=O)ccc([N+](=O)[O-])cc1C c1(C(=O)NCCC(C)NC(=O)C(C)(C)CO)n[nH]c2c1NCCC2 CC1CN(C(=O)Cc2cncc(O)c2)CCC1NC(=O)CCC1CCCOC1 c1(C(N2CCN(C(C34CC(C)(C3)C4)=O)CC2)=O)cccc2cncc(F)c12 CCC1=C(C(=O)NCC2CCCN2C(c2cc3c(C)cccn3c2)=O)CCCO1 C1(C(N(C2CN(C(C3COC(C)(C)CO3)=O)C2)C)=O)COC2(CCC2)C1 c1(NC(C)CSC(F)F)nc(Cl)nc2c(-c3ccccc3)scc12 C1(C(N2CC(CC(C)NC(=O)C(C3CCOCC3)F)C2)=O)C2CCCOC12 N1(C(c2cc(OC)n[nH]2)=O)CCOC2(C1)CN(C(c1ccc3nc[nH]c3c1)=O)C2 C=C(C)C(CC(=O)N1CCC(CNC(c2cnc(OC)nc2)=O)C(C)C1)OCC c1(OC)ccc(O)cc1NC(=O)CN(C(C1CCCOC1C)=O)C(C)C N1(C(C2CC3CC3C2)=O)CCC2(CC1)CC(Nc1ncc3ccnc-3[nH]1)CO2 N(C(=NCC1CCC1)NCC1(CN2CCC2)CCCCC1)Cc1ncn(C)n1 C1(CC)CN(C)CCCN1C(c1cn(C)nc1C)C(=O)NCCCF c1(OC)ncccc1CC(=O)NC(C)CCNC(C1C2CCC1CC2)=O Cc1c(C(=O)NC(C)C(=O)NC(C)Cc2ccnn2C)cccc1O c1(C(N2CCC(=CCNC(C3C(C)C3)=O)CC2)=O)cc2cccnc2o1 N1(C(CC(=C=C)C)=O)CC2CCCC(CNC(=O)C(C)(C)CN(C)C)(C2)C1 CCC(CNC(=O)C(N1CCC(C)(N2CCCCC2)CC1)=O)(CC)CC c1(CCC(=O)N(C)CC2CCN(C(C(C)C3CCC3)=O)C2)cccnc1F n1(CC(=O)N(CCC)CCNC(c2ccc(O)nn2)=O)cnc2c1CCCC2 c1(CNC(C2CCC(n3cc(Cc4ccccc4)nn3)C2)=O)c(Cl)cccc1Cl c1(C(N2CCC(N(C(CC=C)=O)C)CC2)=O)[nH]c(=N)ccc1C Cc1cc(C)c(C(=O)NC(C)CC(C)NC(=O)CC2(O)CCCCCC2)c(C)c1 c1(C(=O)NC(CC)CNC(=O)CC2CCS(=O)(=O)C2)cc(OC)cc([N+](=O)[O-])c1 Cc1ccc(C(=O)NCCC2CCC(NC(c3cccnn3)=O)C2)o1 NC(=O)CCCCC(=O)NC12CC(CNC(c3scnc3C3CC3)=O)(C1)C2 c1(CC(N2CC(F)(C(=O)NCCCCOCC)C2)=O)ccc(Cl)cc1 CCC(CC)CC(=O)N1CCN(C(C2CCCN(C(=O)COCCF)C2)=O)CC1 c1(CC)cc(Br)ccc1C(N1CCCC1CNC(c1ccnn1C(C)C)=O)=O C(=O)(CCC1=CCCCC1)NC1(C)CCCN(C(C2(CCF)CCC2)=O)C1 N1(C(c2cc(C)sn2)=O)CC(NC(=O)C(C)NC(C)(C)C)C(CC(C)(C)C)C1 C1(CC)CN(C(=O)CCC2CCCN2Cc2cc(C)cnc2OC)CC(=O)N1 C#CC1(O)CCN(C(C2(CNC(c3ccc(F)cn3)=O)CCC2)=O)CC1 c1(C(N2CCC(NC(CC(C=C)(C)C)=O)C(O)C2)=O)ccc(F)c(OC)c1F C1(C(N2CCC(O)(CN(C(=O)Cc3ccc(Cl)cn3)C)C2)=O)CC2(C1)CC(O)C2 N1(C(c2n(C(C)C)ncc2)=O)CCC(CNC(C2(C)CCCCO2)=O)C(F)(F)C1 C(CC(CC)C(=O)NC1CCOCC1C(=O)NCC(C)(O)C(F)F)=CC c1(SC)cc(F)ccc1C(=O)NCCCCCNC(C1(O)CCCC1)=O C(=O)(C(O)CCc1ccccc1)NC(C)CNC(=O)Cn1cnc(C(F)(F)F)n1 c1(CC)cccc(C(=O)NC(Cc2ccoc2)C(=O)NC2CN(C(=O)C3CC3)C2)c1 N1(C(CP(C)(C)=O)=O)CCC2(CC1)CN(C(C1CC3CCCCC3O1)=O)CCO2 N1(C(C2(C)CC(C)C2)=O)CCN(C(C2CC(C)CC(=O)N2)=O)CC1C c1(C(=O)NCC2CCC(NC(CC=C=C)=O)C2)cnccc1C(C)(C)C N1(C(Cc2cn(CC)nn2)=O)CC(NC(c2c[nH]cc2C(C)(C)C)=O)CC(F)C1 N1(C(C(C)n2cncn2)=O)CCC2(NC(=O)CCc3ncccn3)CCCC12 c1(CNC(C2CC3CC3N2Cc2cccc(O)c2F)=O)cccc2ccccc12 C(=O)(C(CCN(C)C)NC(C1CC=CC(O)C1)=O)NC(C)Cn1cccn1 N1(C(C2(C)CC(F)(F)C2)=O)CC2(CO)CC1(C(=O)NCCc1cc[nH]n1)C2 C1(S(=O)(=O)NC(C2CCCC2)C2CCC2)(C(=O)OC)CCC1 c1(C(=O)NCC2CC2CNC(C2CC3(CC3)CO2)=O)cc(O)cc(F)c1F C#CCC(C(=O)N1CC(NC(C2CCC(C)CC2)=O)C1)C1CC1 N1(Cc2cc(OC)cc(Br)c2)CCc2[nH]nc(C(=O)NC3COC(=O)C3)c2C1 N1(C(c2cccc(SC)c2)=O)CCC2CN(C(=O)C=CCF)CCC12 n1(CCN(C(C23CSCC2C3)=O)CC)cc(CCC2CCCCO2)nn1 CCCCCCCCCCN(c1cc(NC(C)CC2CCCO2)nc(C)n1)C c1(OC(C(C)CCc2nnc(C)n2C)=O)ccc(F)c(F)c1 CC(C(=O)N(CC(O)CNC(=O)CCC1OCCO1)C)NC(=O)C1CC1 C1(NC(C=CCC)=O)CCC2(CCN(C(C3CCC3c3nc(S)n[nH]3)=O)CC2)C1 N1(C(c2ccccn2)C(=O)NCC(C)C)CCCN(c2nnc(C(C)C)o2)CC1 C1(CC)COC(C)(C)CN1CCNC(c1ccc(C)c(Cl)c1)=O c1(NC(CSCCC)=O)ccc(NC(c2ccc(O)c(C)c2)=O)cc1C c1(CC)c(C(=O)NC2(COC)CCN(C(c3cc(C#N)c[nH]3)=O)C2)cnn1C c1(C(N2CC3CC3(C(=O)NC3CSC3)C2)=O)ccc(Cl)cc1I C1(CC(=O)N(C)Cc2nnc(C)s2)CCCN(C(c2nnc(S)n2C)=O)C1 O=[N+]([O-])c1cccc(C(c2nnnn2C2CCCCC2)NC2C=CCC2)c1 c1(C(=O)NCCN(C(CC(CCC)O)=O)C(C)C)ccc2sccc2c1 C(=O)(CCC(=O)NCC1C(O)C(O)CN1C(=O)CC1CC(=O)NC1=O)NCCC Cc1cc(C(=O)NC2CC(F)CN(C(C3(N(C)C)CCCSC3)=O)C2)cnc1O CCCCCC(F)C(=O)NCC1(C(=O)N(C)Cc2cccnc2)CC12CCC2 C1(NC(=O)Cn2cc(Cl)cn2)(CO)CCCN(C(=O)C(=Cc2c[nH]cn2)F)C1 N1(C(CN(C)C(C2CCN(CCF)CC2)=O)=O)CC2CC(N(C)C)C2C1 N1(C(CCc2cn(C)c3c2cccc3)=O)CC2CC(F)(F)CCC2(C(=O)O)C1 N1(C(CC(COC)C)=O)CC2CCC(NC(=O)CSCc3ccccn3)CC2C1 c1(OC)cc(-c2cccc(C(=O)NCCN3CCN(C)CC3)n2)ccc1[N+](=O)[O-] C(CC(=O)NC1(CO)CN(C(c2cc(=N)[nH]c(Cl)n2)=O)C1)(C(C)C)OCC c1(C(N2CCC(CO)C(O)C2)C(=O)NCc2cccs2)cccc2nc[nH]c12 C1(C(N2C(C(=O)NCC3(F)CN(C)C3)CCC2)=O)CC(F)CN1C N1(C(c2cnc(OC)s2)=O)CC(NC(c2cc(OC)ncn2)=O)CC1(C)C Cn1cc(Cl)cc1CNC(=NCC1CC1)NCC1(C)CCC(=O)N1 CC(C)S(=O)(=NC(=O)c1nn(C)c(Br)c1C)C1CCNC1 c1(CC(=O)N(C(C)CN(C)C(c2cnns2)=O)C)nccn1C c1(OC)cc(OC(F)(F)F)ccc1-c1cccc(C(=O)Nc2cnns2)c1 n1(CCOC)ncc(C(=O)NCCC(O)CNC(C2(COC)CCOC2)=O)c1C C1(C(N(C2CS(=O)(=O)C2(C)C)C)=O)N(C(=O)Cn2cnnc2)CCCC1(C)C c1(OC)ccc(C)c(CNC(C2CCCOC2)=O)n1 N1(C(C2(OC)CCOC2)=O)CCN(C(=O)CCC(C)(F)F)CC1C CC(N=c1[nH]c(=N)[nH]c(=NCC2(N(C)C)CCCOC2)[nH]1)c1nccn1C C1(C2CN(C(C3CCOC3)=O)C2)(NC(=O)C2=C(Cl)CC2)CC1 N1(C(CCN(CC)CC)=O)CCCC1(C(=O)NCc1noc(C(N)=O)n1)CC C(=O)(CC(CC)C(F)F)NCCOCCCN(C(c1c(CCC)onc1C)=O)C CC(C)(O)CCCNC(c1ccc(CN=[N+]=[N-])o1)=O C1(NC(c2nc(CCC)sc2)=O)CCSC12CN(C(C1(C)CC1Br)=O)C2 c1(C(=O)NC2(C)CN(C(COC(C)=O)=O)C2)cc2ccc(C(F)(F)F)cc2nc1O CC(C)C(O)CC(=O)NCCCN1CCN(C(C2C(F)(F)C23CC3)=O)CC1 n1(Cc2ccsc2)nc(CN2CCCC2)nc1-c1cc(COC(F)F)c[nH]1 c1(NC)ccc(C(N2CC(CCCCNC(c3c[nH]nc3C)=O)C2)=O)nc1 CC(C)C(O)CC(=O)NCCC1CCN(C(=O)CC(O)CN(C)C)CC1 N#CC1CCC(C(N2CC(C3(NC(C4CCCC4O)=O)CC3)C2)=O)CC1 N1(C(c2cc(CNC(c3c(C)cc(C)s3)=O)on2)=O)CC(C)C(C)C1C c1(C(=O)NCC2CCCC(CNC(C3(C)C=CCC3)=O)C2)nnc(O)cc1O Cc1cc(Br)c(C(=O)N(CC(C)O)CCNC(C2CC2C)=O)cc1Cl C1(NC(C2CC(C#C)(O)C2)=O)C2CC3C(C2)C13C(N1CC(=O)NC(C)C1)=O C1(C(N(CC(CC)NC(=O)CCC(C)CN(C)C)C)=O)CC2(C1)CC2(F)F c1(C(N(C2CCCN(C(C3C(C)C3)=O)C2)CCO)=O)ccc(S(N)(=O)=O)s1 c1(C(=O)Nc2c(C)n[nH]c2)cc2c3c(ccc2[nH]1)N(C(=O)CCCCCBr)CC3 C1(C(=O)NC2(C)CCCC2)CCC(O)CN1C(=O)CN1CCCCC1 C1(NC(CCC#N)=O)CN(C(C2(c3cccnc3)CCC2)=O)CC1C1CC1 N1(C(CCSCC(=O)OC)=O)CCC(CNC(C23CCC(CC2)O3)=O)C1(C)C CCC(N=c1[nH]c(=NCC2CC(C)(C)C2)[nH]c2ccsc12)c1cc(C)cc(C)c1 N1(C(C2(CC)CC2)=O)CCCC(C2CCN(C(c3cnc(C)[nH]c3=N)=O)C2)C1 N1(C(Cc2n(C)cnc2)=O)CCCCC(CNC(=O)CC2CCC(F)(F)CC2)C1 N1(C(c2c(C)coc2)=O)CC(C)OC2(CCN(C(c3cncc(C)c3Cl)=O)C2)C1 C(CC)(C(=O)N1CCCC1CCC(=O)NCC(O)(C1CC1)C1CC1)OCC N1(C(c2c(NC)nccc2)=O)CCC2(CC2C(=O)NCC(c2cnc[nH]2)C)C1 N1(C(CCOCC(C)C)=O)CCCCC12CC(NC(c1cnnn1C)=O)C2 N1(C(C(C)CC(N)=O)=O)CC2CCCC2(C(N2CCOC(C)(C)C2)=O)C1 c1(NC(CCNC(c2c(C)oc(CO)c2)=O)(C)C)cnc2ccccc2n1 Cc1nn(C(C)C)c(C)c1CC(N1CC(NC(c2ccoc2)=O)C1)=O Cc1ccc(CNC(c2coc(C(C)NC(c3nccnc3C)=O)n2)=O)cc1O C=CC(C)C(C)C(=O)N(CCNC(c1ccc(C)c(NC(C)=O)c1)=O)CCNC C(C(N=[N+]=[N-])C(=O)NC1(CO)CN(C(=O)Cc2cccc(OCC)c2)C1)OCC c1(C(=O)NC(COC(C)=O)C2CC2)cc(C)c2n[nH]cc2c1 N12CC3COCCC3(C1)C2=O.S(=O)(=O)(c1cc(C)sc1C)N1CCN(CC)CC1 Cc1cc(C)c(CNC(C2CCOC2CNC(=O)Cc2cccnc2F)=O)cn1 C1(NC(CC(CCC)C)=O)CCN(C(C2CCCO2)=O)CCC1CO c1(C(N2CC(O)CC(NC(CC3CC(=C)C3)=O)C2)=O)cc2cccc(F)c2o1 C(CC(C(C)(C)C)NC(c1cnn(C(C)C)c1F)=O)N(C(CN(C)CC)=O)C c1(OC)ccc(Br)c(CC(N2CCCC(N3CCCS3(=O)=O)C2)=O)c1 CC1=CCC(NC(C2(C)CCCN2C(C2C3CN(C)CC23)=O)=O)CC1 C1(Nc2oc(C(=O)OCC)c(C(F)(F)F)n2)CCC2C3CCC(C3)C12 c1(C(=O)Nc2c(F)cc(I)cc2F)ccc2c(c1)CCN(Cc1cn[nH]c1)C2 NC1(CO)CCN(C(=O)C(N2CCC(Cc3cccc(F)c3)CC2)=O)C1 Nc1ccc2c(c1)CN(C(=O)C(C1CCC(F)(F)C1)O)CCO2 CCCC(CCCNC(c1cc(C)n(C2CC2)c1C)=O)NC(=O)CC(F)F C1(NC(C(C=C=C)C)=O)CC2CC(C1)N(C(=O)CSc1nncs1)C2 C(CCCC(C)NC(C1CC2CC2C1)=O)NC(Cc1c(C)non1)=O Cc1ccc(C(=O)NC(C(=O)NCC(C)C#N)C2CCCC2)cn1 C12(NC(Cc3c(C)scc3)=O)CC3CCC(C1C2)N3C(C1CCCCC1(F)F)=O C(CCC(=O)N(C1CCN(C(=O)Cc2csc(NC(=O)C(C)(C)C)n2)C1)C)OC C1(NC(CC2(C=C)CC2)=O)CCC(O)CN(C(C2CCN(C(=O)CC)C2)=O)C1 N1(C(C(CCSC)OC)=O)CCCCC2(C1)CN(C(=O)Cn1ncnn1)C2 C(CC1CC1)(CC(=O)NCC(C)CCCO)NC(c1cc(C(C)=O)[nH]n1)=O c1(CCC)nc(C(=O)N(CCCNC(=O)C(C)c2ccon2)C(C)C)cs1 N1(C(C(C)OCCCC)=O)CCC2(CC1)CC2C(N1CCn2nccc2C1)=O C#Cc1ccc(CNC(C2(C(C)NC(C3CC4CCCC4C3)=O)CC2)=O)cc1 N1(C(CN(C)C)=O)CC2(CCOCC2)CC1CNC(=O)C(C)(C)C1CCOC1 Cc1cc(NC(C2CCN(C(=O)C(O)C3CCCC3)CCO2)=O)cc(C)c1F C(C(CC)(CC)C(=O)N(C1CCC2CC12)C)NC(c1c(CC)n[nH]c1)=O C1(NC(C2CC(C)(C)C2C(F)(F)F)=O)CC(F)CN(C(=O)Cc2cc[nH]n2)C1 N1(C(CCc2cc(C)oc2C)=O)CCN(C(C2C=CCC2)=O)C2(CC2)C1 c1(C(=O)NC2C(CNC(=O)CSC3CC3)CCC2)ccc([N+](=O)[O-])s1 CCCCCC(C)CC(=O)NCC(C)(CO)NC(c1cnc(C)[nH]c1=N)=O c1(NC(N2C(C3(O)CN(C(c4c(C)nsc4)=O)C3)CCC2)=O)occ2c1CCC2 Cc1cc(CC(=O)NC2CC(F)(CNC(C3COC(=O)C3)=O)C2)cc(C)c1 c1(C(=O)NCC(=O)NC(CC)CNC(=O)C(N)=O)ccc(OC)cc1 N1(C(C(C(C)C)CNC(C2CCOCC2(C)C)=O)=O)CC2(C)CC1CCO2 C(C1CCCN1C)=CC(N1C(C2(NC(CN(CCC#C)C)=O)CC2)CCC1)=O C(=O)(CCC(C)SC)NCCCN(C(C(C)OCC=C)=O)C(C)C C(=O)(CC1=CCCC1)N(C1CN(C(=O)COC2CC2)CC12CC2)C C=CCCCC(C)(C)C(=O)N1CCCC1CN(C)C(C1CCC(C)(C)OC1)=O CC1(C(=O)Nc2ccccc2)CC(=O)CC(C)O1.C12CCN(C1)C2=O N1(C(=O)COC2CCCC2)CC2(C1)CN(C(C1CCC3(CCC3)O1)=O)CC2CO C(=O)(C(C)=Cn1ccnn1)N(CC(N1CCN(C(C(CCC)(C)O)=O)CC1)=O)C N1(C(CN(C(C2C(C)SCCC2)=O)CC2CC2)=O)CCC(C)(O)C(O)C1 C1(CNC(c2nccc(OC)c2)=O)CCN(C(C2CCCC23CC3)=O)C12CCC2 C(=O)(C1=C(C)CCC1)NCC(=C)CCNC(C1CC(C)N1C(=O)OC(C)(C)C)=O CN1CCCCC1C(=O)NCC=CCC(=O)NCCC(O)C1CC1 C1(c2ccccc2)(CC)CCCN(C(=O)CCCCCNc2oc(Br)nc2C)C1 N1(C(C2(CC)CCCN2C(=O)C=C2CCC2)=O)CCc2nn[nH]c2C1 C(C(CCO)NC(C1CCCC1NC(=O)C=CCO)=O)N(C)C N1(C(CCc2ccc(OC)cc2)=O)CCC2C(CCCN2C(=O)C(C)C(C)C)C1 c1(C(=O)NCC(C)(CNC(C2CCCC2O)=O)OC)ccccc1SC c1(C(=O)NCC2CC(CNC(c3nc(SC)oc3)=O)OC2)cc(OC)ccn1 N1(C(CNC(=O)OC)=O)CCC(C(=O)NOCc2cccc(F)c2)(OC)C1 C1(NC(Cc2cc(OC)no2)=O)CCCN(C(=O)C=Cc2cccc(F)c2)CC1 C1(C2CCC(CCCC)CC2)NC(=O)N(CC)C2=C1C(=O)NC2c1ccccc1 C(=O)(C1CCCc2cncn21)N(C1CN(C(c2c(CC)nn[nH]2)=O)CC1(C)C)C c1(C(=O)NC2CCC(CNC(c3c(C)nc(N)cn3)=O)C2)cc(F)c(F)cc1F c1(-n2cc(C(=O)NCC34CC(NC(CC=C=C)=O)(C3)C4)nc2)ccc(Br)cc1 c1(OC)ccnc(C(=O)NCC(C)(C(C)C)NC(=O)Cc2cn(C)nn2)c1OC CC(C)C(C(=O)N1CCCCCO1)C(C)NC(C1CN(C2CCC2)C1)=O C1(CC)CCN(C(=O)Cc2nocc2C)C1C(N1CC[Si](C)(C)C1)=O C12(C(=O)Nc3scc(-c4cn(C(CC=C)CC=C)nn4)c3)CCCN(CCC1)C2 C1(C(N(CC(=O)NC(C#C)CC2CC2)CC2CC2)=O)CC2CC(=O)C1O2 N1(C(c2c(C#C)c[nH]n2)=O)CCC(C2(NC(c3cc(CC(C)C)[nH]n3)=O)CC2)C1 c1(C(c2nnnn2CC)NC(CCCC=C)C2CC2)csc(S(N)(=O)=O)c1 Cc1cc(C(c2nnnn2CCCF)NC2CC(Cn3ccnc3)C2)no1 c1(C(C)C)ccc(C=CC(N2CCCC(NC(C3(C)CC4CC4C3)=O)C2)=O)cc1 C1(NC(CC(C)(O)C2CC2)=O)CN(C(=O)C#CC2(C)CCCO2)C2CCCCC12 C1(CNC(=O)COCCc2cccs2)CCCCC1NC(c1ccnc(Cl)c1)=O C12(C(N3CCCCC(C(=O)NCC45CCC(CC4O)C5)C3)=O)CCN(CC1)CC2 N1(C(=O)CCNC2(CF)CC2)CCOCC1c1cccs1 C12(CNC(CSCC=C)=O)CCC(CNC(c3ccc(C)c(C)n3)=O)(CC1)OC2 c1(C(=O)NCC(C)NC(C2CC(=O)N(C)C2)=O)cc(F)ccc1Cl CCC1=C(C(=O)NCC(C2CC2)NC(=O)CCc2csc(C)n2)SCCO1 CC(CO)CCCNC(=O)C(F)CC1CN(C(C2CN(C3CCC3)C2)=O)C1 C1(C)(C(=O)NCC(CC)NC(=O)CCC2CCCN(C)C2)CC(=O)N(C)C1 c1(CSCC)ccc(CC(=O)N(CCCNC(c2nncs2)=O)CCO)cc1 c1(C(N(C2CCCN(C(CCSCC(C)C)=O)CC2)C)=O)ccc(Cl)c(F)c1F c1(C(N2CCC(N(CCO)C(c3cnc(O)s3)=O)C2)=O)cc2cccnc2o1 CCC(CNC(=O)CCc1cccc(C)c1)(CC)NC(=O)CC1CCCC(=O)N1 C1(NC(C2CC3(CCC3O)C2)=O)CCCCCC1C(=O)NC1COCCOC1 C1(C(=O)Nc2c(C(=O)NC(Cc3ccc(C)s3)C)n[nH]c2)CCC(F)(F)C1 N1(C(c2ccc(SC)o2)=O)CCC2CCN(C(c3ccn4nnnc4c3)=O)CC12 C1(NC(CCc2ccc(CC)cc2)=O)CS(=O)(=O)CC1NC(c1nnn(C)n1)=O C(=O)(C(Cc1ccccc1)N(C)C)NC(C)CCNC(C1(C(C)(F)F)CCC1)=O c1(C(=O)NCC(CC=C)NC(c2n[nH]cc2C2CC2)=O)nn(C)c(=O)cc1C c1(CC)ccccc1N(C(=O)COC1CCN(C(=O)C=CC(F)F)C1)C C=C=C(C)CC(=O)NC1CN(C(C23CSCC2C3)=O)CC1SC CC1(C)CCN(C(C2CN3CCC2CC3)=O)C(C(=O)NC2CNC(=O)OC2)C1 CC1CC2(CCN(C(=O)CC3NC(=O)NC3=O)CC2)CN1C(=O)C(Cl)=CCl Cc1cnc2ccc(C(=O)N(C(C)CNC(=O)Cc3ccon3)C)cn12 C=Cn1nccc1C(=O)NCC(C1CCCC1)NC(C1CC(N=[N+]=[N-])C1)=O c1(NC(C2CCN(C(=O)C=CI)C2)C)cnc(C#N)cn1 Cc1cc(C(N2CC3CCC(C2)C3NC(c2cnc(C)[nH]2)=O)=O)c(F)c(F)c1 Cc1nc(CN2CCC(C(=O)Nc3cc(O)ncc3C)C(O)C2)ccc1Br c1(C(=O)NCCCOCCN(C)C(c2cscn2)=O)cnc(N)c([N+](=O)[O-])c1 N1(C(c2c(C)ccs2)=O)Cc2n[nH]cc2C1C(=O)NCC1(CC2CC2)CC1 c1(OCC(=O)NCC2(CNC(C3C4CCCOC34)=O)CCC2)ccc(F)cc1F c1(C(N2CCN(C(CNC(C3N(CC)CCC3)=O)=O)CC2)=O)cccc(F)c1N c1(CNC(C(CSC)NC(=O)CC2CCC(=O)N2)=O)oc(C)nc1C C1(NC(C2CCCC23CCC3)=O)CC2(CCN(C(c3cc4cscc4s3)=O)C2)C1 N1(C(C(=Cc2cccnc2)C)=O)CCC2CN(C(C3CCC3(C)C)=O)CC12 N1(C(C(C)SCC)=O)CCC2(CC1)OCCCC2NC(=O)C#CC(=O)N(C)C C(c1cccc(O)c1)=CC(N1CCCC(CNC(C2N(C)CCC2)=O)C1)=O C1(c2n(CC=C)nnn2)(NCC2CC(F)C2)CCN(c2ccncc2)CC1 c1(NC(C2N(C(C(CC(C)C)O)=O)CCCC2)=O)ccc2[nH]ccc2n1 C1(CC=C)(NC(=O)C=NOC)CCCN(C(C2CCCCNC2=O)=O)C1 C(=O)(CCCCCC#N)NC(C1(CNC(c2cccnc2)=O)CC1)C C1(C(=O)NCC2N(C(C(C)=C(CC)C)=O)CC2)CC2CC1C1C2C1(F)F C(=O)(CCCCCC)NC(C1(CNC(C(C)OCC=C)=O)CC1)C c1(C(N2CC(O)(C(C)NC(C3CC(Cl)(Cl)C3)=O)C2)=O)c(Cl)ccc(Cl)c1O c1(C(N2CCC(F)(CO)CC2)=O)c(O)ccc(F)c1F.C12CC1CNC2=O C1(C(=O)NCc2nc(C)[nH]n2)(NC(=O)C=CCCC(C)C)CCC(C)(C)C1 c1(CC(=O)NC2C(C)CCN(C(=O)Cc3ccon3)C2)ccc2c(c1)CCCC2 C1(CC(=O)NC(C)CC(F)(F)F)N(C(=O)OC(C)(C)C)CCC1(C)C Cc1ccc2c(c1)SC(C(N1CCC(C3(NC(c4ncn(C)n4)=O)CC3)C1)=O)C2 O=S(=O)(c1cccc(=NC2CC2C2CCOCC2)[nH]1)NC1CCOCC12CCCC2 C1(OCC)CC2CN(C(=O)CC3CC(C)N(C(=O)C(C)C(F)F)C3)CC12 C(CCN(C(=O)CCc1ccc(F)cc1)C)(C(C)C)NC(c1cn(CC)nc1)=O CCCC(CC)NC(C)COCC1CC1.C(COC)O CC1CC(N(C(=O)CN(C2CCC2)C)C(C2(O)CCOCC2)=O)CC(C)C1 CC1(C)CC(Cn2ccnn2)CN1C(c1ccc(Nc2cccc(F)c2)o1)=O Cc1cc(C#N)ccc1C(N1CCC(CF)(NC(c2cccc(CF)c2)=O)C1)=O CC1CCCCC1C(=O)NC1CCN(C(c2cnc(-c3ccoc3)s2)=O)C1C C=C(C)CC(C(=O)NC(C(=O)NCC1CCC(=C)CC1)C1CC1)OC c1(C(=O)NC(CNC(CC(C=C)C)=O)CO)cc(S(N)(=O)=O)ccc1Br C1(C(=O)OC)CC2(CC(NC(=O)NC(c3cccc(F)c3OC)C(F)(F)F)C2)C1 c1(C(N2CC3CC3(NC(C3(CO)CCCO3)=O)C2)=O)cnc(C2CC2)nc1 N1(C(c2c(CCC)n(C)nc2)=O)CCN(C(C2COCC(C)O2)=O)C2(CC2)C1 CCCCC(C)C(=O)NC(C)CNC(c1ccccc1-n1cc(Br)cn1)=O C12(NC(C(CC#C)O)=O)CCCC1(F)CN(C(c1cnc(C3OCCO3)s1)=O)C2 C1(OC)(CNC(C2CC2F)=O)CCN(C(c2oc(CO)nc2C)=O)CC1 c1(C(=O)NCC(C)(CNC(=O)CC2CC3CC3C2)OCC)cc(C(C)C)oc1C CC1(C)CC(C(=O)NCC2COC(CN=c3cc(C(N)=O)nc(Cl)[nH]3)C2)=NO1 c1(CN2CCC(OCc3cn(-c4cccc(N)c4)nn3)CC2)ccc(F)c(Br)c1 C12(OC)CCCCC(C(=O)NC3(CNC(C4CCCS4)=O)CCOCC3)(C1)C2 c1(NC2CC(NC(C3CCCN3C(c3ccccc3)=O)=O)C2)ccc(O)cn1 c1(C(N2CC=CC(NC(CN(C3CCSC3)C)=O)C2)=O)cc2c(nn1)CCCC2 C(=O)(CC(C)CC(=O)NCC1(C)CCC(NC(c2cnc(C)cn2)=O)CC1)OC Cc1noc(CNC(=O)CC2CCCN2C(=O)CN(C2CCCC2)C)n1 C1(CNC(C2(C(=O)OCC)CCC2)=O)C(C)CCCN1C(=O)C1=CSCCO1 C1(C(=O)NCC2(CCNC(C(C3CCC3)OC)=O)CC2)CCCN1C(C)C C1(NC(CCC2(C)CC2(F)F)=O)CC(NC(=O)COc2cccnc2)C12CCC2 c1(C(=O)NCC(C)CNC(=O)CCC2CCCCO2)cccc2c[nH]nc12 N1(C(CC(C)C(C)(C)NC(C2CCCO2)=O)=O)CCC2(CNC(=O)N2)C1 C1(N(C(CC)=O)CSc2ccccn2)CCCN(C(=O)Cn2ccnc2C)CC1 C(=O)(C(F)(F)C(C)(C)O)NC1CC(C(=O)NC(c2ccccn2)C)C1 C#CCCCC(C)C(=O)NC1CC(C)(NC(=O)CCCc2ccc(O)cc2)C1 C(=O)(C(F)CC(C)(C)NC(=O)COc1ccsn1)NC1CC(C)(CC)C1 C1(C(=O)OC)CN(C(c2ccc(C(F)(F)F)nc2OC)=O)C2(CCCC2)C1 c1(OC)ccc(Cl)cc1C(=O)N(c1ncccn1)CC1(C)CCNCC1 c1(OC)c(C(=O)NCC2CCCC(NC(=O)C(C)(C)CO)C2)csc1Cl c1(CC(C)C)ccc(CC(=O)NC2CC2NC(C2(C#N)CCC2)=O)cc1 c1(C2CN(CC)C2)cc(OC)c(OC)cc1Br.C1C(C(C)C)CNC(=O)N1 C1(CCC)CN(C(=O)C(CC)SC)CC1C(=O)NCc1cccc(C)n1 CC1CC(C(=O)NCCn2cc(CO)nn2)CCN1C(C1OCCOC1C)=O Cc1cc(C(=O)NNC(=O)N(CCCO)CCCO)cc([N+](=O)[O-])c1Cl c1(CC(N2C(CNC(c3cnncc3O)=O)CCCC2)=O)ccc2n[nH]cc2c1 C1(NC(C(CCSC)O)=O)CC(F)(F)CC1NC(c1snnc1C(C)C)=O C1(C(N2CC3C(CNC(C4C(C(=O)OC)C4)=O)(CC3)C2)=O)C2CCC3C(C2)CC13 Cc1ccnc2c(C(N3CC(CNC(c4ccnnc4)=O)CC3(C)C)=O)cnn12 CC1(CNC(c2ccsc2)=O)CCN(C(C2CCCN2c2ccccc2)=O)C1 C(N=c1[nH]c(Cl)nc2[nH]ccc12)C1OCCN(C(c2cc(Br)co2)=O)C1 c1(C(=O)NC)ccc(C(N2CCCC2CNC(=O)C=Cc2cc[nH]n2)=O)cc1F c1(C(N2CCC(C)(CNC(C3CC4OC3C3CC43)=O)C2)=O)c(F)cc(Cl)cc1F C1(S(C)(=O)=O)(C(=O)Nc2scc(-c3c(F)ccc(C(=O)NC)c3)c2)CCCCC1 Cc1noc(N)c1C(=O)NC1CCC1NC(c1ccnnc1)=O c1(CC)noc(CCC(N2CCCC2CN(C(=O)C=CI)CC)=O)n1 C1(CNC(CSCCN(C)C)=O)(NC(C2CCCO2)=O)CCOCC1 c1(C(=O)NCC2CN(C(c3scc(OC)c3)=O)C(C)CC2)ccc(F)c(C#N)c1 C#CC(C)(C)C(=O)N(C1CC(NC(c2nccnc2C)=O)C1)C C1(C(=O)NCCC(c2cccnc2)N(C)C)CC1C1CCC1 C1(C(N2CCC(N(C(c3cc(O)n(C)n3)=O)CC)C2)=O)CCC(C2CC2)C1 C1(CC)CN(C(C2CN(CC(F)(F)F)C2)=O)CCC1NC(c1cc[nH]c(=N)c1)=O C1(C(=O)NCc2c(C)nccn2)CC2C=CC1N(C(c1ocnc1C(C)C)=O)C2 C#Cc1cccc(C(=O)NC2CCC(N(C)C(c3cncnc3C)=O)C2)c1F CN1CCOCC1C(=O)NC1CN(C(C2CSC2)=O)CC1CC(C)(C)C C1(CNC(C2CC(CC3CC3)C2)=O)CN(C(C2(C3CCC3)CC2)=O)C2(CCC2)C1 C(=O)(C1=CC2CCC(C1)C2)N1CC(NC(C=COCC)=O)(COC)C1 N1(CC(=O)NCC(CC(F)(F)F)NC(c2ccc(O)cn2)=O)C(=O)CCCC1=O c1(C(N2C(C(=O)OC)CC(n3cc(C(C)O)nn3)C2)=O)ccc(Br)cc1[N+](=O)[O-] N1(C(C(CCC)NC(N)=O)=O)C2CCC1CN(C(C1CC1(C)CC)=O)CC2 C1(COC)(NC(=O)C2CC2)CCN(C(C2(c3cccc(C#N)c3)CC2)=O)CC1 C1(NC(C(C)(C)OC)=O)CC2CC1CN2C(c1cnn(C2CCCCC2)c1)=O N(C1CCc2c(C(=O)O)cccc21)CC(CC)C#N C1(OC)CCC(CC(=O)NC2CCN(C(C3CN(C4CCOC4)C3)=O)C2C)CC1 N1(C(C(CCNC(c2c(CC)csc2)=O)O)=O)CCCC(OC)C1C c1(C(=O)NCC2C3CN(C(C(CC)O)=O)CC32)ccc(=NC)[nH]c1 C(=O)(C(F)C(C)C(F)(F)F)N1CCN(C(Cc2ccc(SC)cc2)=O)C(C)C1 C1(C(=O)NC2(CNC(c3nccc(N(C)C)c3)=O)CCC2)CC2(CCCC2)CO1 C1(C(=O)NCC2C3CN(C(c4ccc(C#N)[nH]4)=O)C2C3)CCC=CCCC1 C(Cn1cccn1)(C(=O)NCc1ncon1)NC(=O)CCc1cscn1 c12cccc(c1)CNCC2N(c1cc(C)sc1)C.c1(C(C)(C)C)c(C)noc1Cl C1(C(=O)NCC2(F)CN(C(CN(C)C(=O)C3CC3)=O)C2)C2CC3CC(C2)CC1C3 CCC(=O)CCC(=O)N1CC2(CC2)CC1C(N1CCC2C(C(N)=O)C2C1)=O Cc1cc(=NC(C)C2CCN(C(c3cn4cc(Cl)cnc4n3)=O)C2)[nH]c(C)n1 N1(C(C)C)CCC(C(=O)NCC2CC2CNC(c2occc2C(C)C)=O)C1 c1(C(=O)NCC(C2CC2)NC(=O)C=CC2CC2)nc(C2CC2)cs1 N1(C(c2c(CC)n(C)nn2)=O)CC(NC(=O)C(C)OCC(C)C)CC1(CC)CC C1(CNC(c2c(C)nc(O)[nH]2)=O)CCN(C(=O)Cn2cnc(C#N)n2)CC1(F)F Cc1nc(NC(C2CC(F)CN(C(c3csc(Br)c3)=O)C2)=O)ccc1C(F)(F)F N1(CC(=O)NCC(c2ccccc2)NC(c2ccc(C)[nH]2)=O)OC(C)(C)CC1=O n1(CC=C)ccc(CN(C(N2CCSCC2)=O)CC)n1 n1(CC(=O)OC)ccc(=NC(=O)CNC(=O)C(C)N=[N+]=[N-])[nH]1 N1(C(CNC(CC)=O)=O)CCC(C)C(CNC(C2CCCCN2C(=O)CC)=O)C1 c1(C(N(CCCNC(c2cccc(CC)n2)=O)CC)=O)cccc2cncn12 N1(C(Cc2ccc(C(N)=O)cc2)=O)CC2CC(C1)CN(C(=O)Cc1cncs1)C2 C1(C)C(=O)N(CC)CC(CO)NC(=O)O1.C(C)(=O)OCC CCC(CO)C(=O)NCCN(CCOC)C(c1cc(-c2ccccc2)[nH]c1C)=O c1(C(N(CCCNC(CC(C)C(F)F)=O)C)=O)c(O)ncc2c1CCC2 CC1CN(C(c2cnn[nH]2)=O)CC1CNC(=O)C(c1cccc(Cl)c1)(C)C C(CC(C)C(=O)NC1CN(C(=O)Cc2cnns2)CC1OC)=CCC c1(CSCC)ccc(C(=O)NC2CCC(NC(=O)C(C)c3ncco3)CC2)cc1 O=C(C(O)C(F)F)NCCCCC1CN(C(c2ccc(C3(F)COC3)cc2)=O)C1 N1(C(C(C(C)C)NC(C2(C)CCCC2O)=O)=O)CCN2CC(C)CC2C1 c1(N2C3CN(C(C(C(C)C)O)=O)C(C3)C2)nc(Cl)nc2cnn(C)c12 C#CCCC(C(=O)O)NC(=O)C(C(C)OC)Oc1ccccc1Br C1(N(C(=O)C(Cl)=CCl)C)CCC(NC(=O)CN2CCS(=O)CC2)CC1 c1(C(N(CCOC)C(C)C2CC2)=O)cc(=O)n(C)cn1.C(=O)(C(F)CC1CC1)N c1(OC)ccc(Br)cc1C(N1CC2CC2(CNC(c2cnn[nH]2)=O)C1)=O c1(CC)ncc(C(=O)N(C)CCc2ccccc2C(C)(C)C)c(=O)[nH]1 C(C(=O)N=c1cc2n([nH]1)CC(C)OC2)Oc1c(CC)nc(C)cc1 C1(NC(=O)CCC2CCCCCC2)CN(C(=O)C=C2CCC2)CC12CCC2 CC1CCCC(C(=O)N(CC(=O)N(C2(C3CC3)CC2)C)C)CC1 N1(C(C2(COCC)CC2)=O)CCOC2(CCN(C(=O)CC(C)n3cccc3)C2)C1 C1(C(N(C2CCN(C(c3cnn(C4CC4)c3)=O)C2)CC)=O)CC2(CCO1)CC2 C(=O)(CS(=O)(=O)C1CCCC1)N1CC(N(C(c2csc(C)c2N)=O)C)C2(C1)CC2 C(CC(C(=O)NC1CN(C(N)=O)C1)NC(c1cn(CC)nn1)=O)=CC Cn1cncc1C=CC(N1CCCC(CCNC(C2CC2c2ccsc2)=O)C1)=O N1(C(Cc2c(OC)cccc2)=O)CC2CCC1CN2C(c1cc(=O)cc(Cl)[nH]1)=O C1(C(N2CC3N(C(C4C(CCOC)C4)=O)C(C3)C2)=O)CC2CCCC(C1)C2 C1(C(=O)NC(CNC(c2c(SC)nn(C)c2)=O)C(C)C)CCN(C)C(=O)C1 c1(C(=O)NCCC(C)NC(CSCC)=O)[nH]c(C)c(C(C)=O)c1C CC1(C)COCC(C(=O)NCC2(C)CCN(C(C3CC=CCC3)=O)C2)O1 c1(COC(C=COCC)=O)ccc(C)cc1.C1C=CCN1 c1(N(CC)CC2(C3CCC3)CC2)cc(C)cc(F)c1 N1(C(CCCC#N)=O)CCC2CN(C(=O)C=Cc3ccc(F)cc3)CCC2C1 CC(CNC(=O)CC1(O)CCOC1)CC(=O)NCC1CC2(CC2)C1 C(CC(C(=O)N1CCCC(C)C1)NC(=O)COCc1nc[nH]n1)=CC N#Cc1cccc2c1CCN(c1nc(C(F)F)ns1)C2 c1(C(=O)NCC(CN(C(CCCC(=O)OC)=O)C)C)cc2nnn(C)c2s1 C(CC1=CCN(C(=O)Cc2cc(F)cc(F)c2)CC1)NC(c1cc(C)ncn1)=O C(=O)(CCCCCCN=[N+]=[N-])NCC1N(C(C(C)=C(CC)C)=O)CC=C1 C1(NC(CN(S(C)(=O)=O)C)=O)CCC(NC(=O)C(F)n2cccn2)CC1 c1(C(=O)NCC2CN(C(C(CCSC)(C)C)=O)C2)cc2cc(C)ccc2o1 c1(-c2ccc(C(N(CCOC)CCNC(=O)CN3CC=CC3)=O)s2)cccc(C)c1 N1(C(CC(CC)C2CC2)=O)CC(CNC(=O)C=Cc2ccc(C)s2)C2(CC2)C1 CC(C)C(O)C(=O)NC(CNC(=O)C(C)C1CCCO1)C(C)(C)C C(C(CC(=O)N1CC2CC1C2CO)OC)NC(CNC(=O)OCC=C)=O C=CCCCCCC(=O)N1CC(C(=O)NOC(C)C=C)C2(CC2)C1 Cc1nnc2n1CCC2(C)C(=O)NC(C)CNC(=O)C(C)(O)C(F)(F)F Cc1ccc(Cl)c2[nH]c(C(N3CCC(CNC(=O)CC(C)C)C(C)C3)=O)cc12 N12CCC(C13CCCC3)C2.Cc1cccc(C2CCCCC2NCC(=O)OCC)c1 C1(C(=O)Nc2cnoc2)CSCCN1C(c1cncc(F)c1)=O C1(CNC(Cc2n(C)cnn2)=O)CC2COCC2N1C(=O)C1=COCCC1 C1(NC(=O)NC2(CC)CCCC2)CCCN(C(c2cccs2)=O)C1 c1(OC)cc(C)c(C(N2CC(NC(c3ccccc3)=O)C(F)(F)C2)=O)cn1 C1(C(=O)NC2CCN(Cc3cnn[nH]3)C2)(CO)CCOCC1 Cc1oc(Br)cc1C(=O)NCCC(C)CCNC(c1nn[nH]c1C)=O c1(N(C)C)nc(C(N2CCCC2CNC(c2cncc(N)c2)=O)=O)cc(O)n1 N1(C(c2ccn(CC(C)C)n2)=O)CC(C)CCC1CNC(c1cnc[nH]c1=N)=O C1(C2CCN(C(=O)CCC(C)(C)F)C2)(NC(C2N(C(C)=O)CCC2)=O)CC1 c1(N2C3(CN(C(c4ccc(OCC)nn4)=O)C3)CC2)ncnn2cc(Br)cc12 N(C(=NCC1=CCCC1)NC(C)C1CC1)C1CCC(NCC(C)C)CC1 c1(C(=O)NC2CC(N(C(=O)CC3C=CCCC3)C)C2)coc2c1C(=O)NCC2 CC(CCC(=O)NCC(F)C(C)(C)O)NC(c1c[nH]c(=N)o1)=O C(CN=c1[nH]c(C)nc2[nH]ccc12)c1ccc(CNC(CC)=O)c(F)c1 CN1CCN(C(=O)Cc2cc(O)nnc2O)C(CNC(C2CCSC2)=O)C1 C1(C#N)(C(N(C2CCN(C(C(CC)OCC)=O)C2)CCO)=O)CCCC1 CC1CCN(C(=O)C=CC(=O)N(C)C)CCN1C(=O)C=CC(=O)C1CC1 c1(C(=O)NCCCC(=O)N(CC(O)CNC(=O)CSC2CC2)C)ccc(O)cc1 C12(NC(c3n[nH]c(C)c3Br)=O)CCC1CN(C(=O)C(O)CCN(C)C)C2 c1(C(N2CCC(N(CC(C)C)CCC)CC2)=O)cnn2ccccc12 S(=O)(=O)(c1ccc2c(N)cccc2c1)N1CCC(C(N2C(CC)CCC2)=O)C1 C1(CCN(C)C)CCN(C(=O)C(c2ccccc2)N2CCOCC2)C1 Cc1cnc2nc(NC(=O)NNC(=O)c3cnn(CCN4CCOCC4)c3)sc2n1 N1(C(C2CC(NC(C(CSC)C)=O)C2)=O)CC2(C)CC1CCO2 C=CC(CC)C(=O)NCCCN(CCCNC(C1C(C(C)=O)C1(C)C)=O)C c1(NCCC(C(=O)N(C)C)(C)C)cccc2nnn(C)c12 CC1Cc2cc(C(=O)NCC3CCCN3C(C3(CCF)CC3)=O)ccc2O1 C1(CC)(NC(c2cc(C)c(C)s2)=O)CCN(C(=O)Cc2conc2C)CC1 C1(NC(CN(C(Cn2ncc(CC)c2)=O)C(C)C)=O)CC2(C1)CC(C)(C)C2 N1(C(C=CCC)=O)CCc2nc[nH]c2C12CCN(C(C1CC(N(C)C)C1)=O)C2 N1(C(C=CC2CCN(C(C(C)C3CC3)=O)CC2)=O)CC(O)C(O)C12CCC2 c1(C(N2CCOCC(CNC(=O)C=CC3CC3)C2)=O)cc2c(O)ncnc2cn1 c1(SC(C)CCNC(C2CCC(C(=O)OC(C)(C)C)C2)=O)cnn2cccc2c1 CC(C(=O)NC1CC2CC(NC(c3csc(Br)n3)=O)CC12)C(C)(C)O Cc1cnc2nc(C(N3CCC(C)C(CNC(c4cccnc4)=O)C3)=O)nn2c1 C1(CNC(C2(C)CC=CCC2)=O)CN(C(=O)C(F)=C2CCC2)CC12CC2 Cc1ccc(C(=O)NCC(CNC(=O)CNS(N)(=O)=O)C(F)(F)F)cc1[N+](=O)[O-] CC1CN(C(=O)COCC2CCCCO2)CC1CNC(C1CC(C)(F)C1)=O c1(-c2n(CC=C)nc(-c3cc(F)cc(Br)c3)n2)cc(OC)c(OC)cc1OC CCC(C(=O)NCc1cc(C)c(C(=O)NC(CO)CCC)o1)C(C)C Cc1ccc(Br)c(CCC(=O)Nc2ccc(Br)c(Br)c2)c1 C1(NC(C=C(CC)CC)=O)C2COCC1CN(C(c1ccc(Cl)c(Cl)c1)=O)C2 C12(C(=O)NC(C(CO)SC)C)C(=O)C3CC1C2C3.C1(=O)C2=NOC(C2)CN1 C1(NC(c2c(OC)n[nH]c2)=O)CCCC(NC(=O)C(CCSC)OC)C1 C1(NC(C(C2CCOC2)NC(c2ccc(CO)o2)=O)=O)CCN(CCO)CC1 Cc1c(Br)c(C(N2CCCCC2CN(C)C(C2(F)CC=CC2)=O)=O)nn1C C1(C)(C(N2C(CC)CCC2)=O)CC(O)CN1C(=O)COc1ccccc1 N1(C(c2cc(CCC)[nH]n2)=O)CCCC(CCNC(=O)C2=C(C)CCC2)CC1 S(=O)(=O)(c1ccc(F)c(Br)c1)N1CC2CN(C(=O)Nc3cc(C)cc(C)c3)CC21 N1(C(c2c(OC)ccs2)=O)CC(C(=O)N(C(C)C(C)(C)C)C)C2(CC2)C1 C1(C(=O)NC2CC(CCNC(C=CC(=O)N(C)C)=O)C2)CS(=O)(=O)CC12CC2 C1(C(=O)NC(CCC=C)C)CC(O)CN1C(=O)CN1CCCCC1C N1(C(c2cc(C)c(CO)cn2)=O)CC2CCC(C1)C2NC(=O)C(C)C(C)(C)C c1(CC(=O)N(CC(CC)NC(c2cc(OC)nn2C)=O)C)c(Cl)cnn1C Cc1ccc(C=CC(=O)NC2CC(C)N(C(=O)Cc3cnns3)C2)cc1 C1(C2CN(C(c3ccc(Cl)c(OC)c3)=O)C2)(NC(c2ccc(CC)cn2)=O)CC1 C1(C(N2CCC(N(C(=O)C(C)(C)c3cccnc3)CC)C2)=O)CCCC(OC)C1 N1(C(C(C)NC(=O)C2CC2)=O)CCOCC1CCNC(C1(C)CCC(=O)N1)=O Cc1scc(C(=O)NC2CC(CNC(c3cc(C4CC4)ns3)=O)C2(C)C)c1C c1(C(N2CCC(CO)(Nc3ncccn3)CC2)=O)ccc2nncn2c1 C1(O)(C(=O)NCC2N(C(C(F)=CC)=O)CC2)CCSCC1 c1(C(N2CC(C)OC(CCNC(=O)C(F)=CCCF)C2)=O)ccc(N)c(F)c1F c1(C(=O)NCC2N(C(C(COCC)C)=O)CC(O)C2)c(F)ccc(O)c1F C1(OCC)(CNC(C2CC=CCO2)=O)CN(C(=O)CCNC(=O)COC)C1 Nc1nc(Cl)ccc1C(=O)NCCC1CCN(C(=O)C(C2CCCCC2)O)C1 N#Cc1ccc(=NCC(=O)NC(CNC(c2n[nH]c(O)n2)=O)C2CC2)[nH]c1 C1(NC2(c3n(CC(=O)OC)nnn3)CCSC2)CCOC(c2ccccn2)C1 Cc1nc(C(=O)Nc2nnc(-c3ccc(C)n3C)s2)nn1-c1cccc(F)c1 c1(N2CCN(C3CCN(C(c4nnn(CC)c4C)=O)C3)CC2)cnc(C#N)cn1 N1(CC(=O)N(C)CC=CC(=O)NC(C)C)CCCCC1C.c12cncc(c1)OCCC2 n1(CC(=O)NC23CN(C(c4c(COC)nn[nH]4)=O)C(C2)C3)cc(C)ccc1=O C1(C(=O)NC2C(C(=O)NCCCn3ncc(C)c3)CCC=C2)CC2CC(=O)C1O2 C12(NC(C(C)(C)c3cccnc3)=O)COC(CNC(c3scnc3Cl)=O)(C1)C2 c1(OCCC)ccc(CC(=O)OCC)c(OC)c1.C12(C)CCN1C2=O c1(C(N2C(CNC(C3COCCO3)=O)CC2)=O)cccnc1S C#CCC(CC(=O)NCCCN(C)OC)NC(=O)CC1CC(CC)=NO1 Clc1ccccc1-n1nc(Cn2cc(Cl)cn2)nc1Cn1nnc(-c2ccco2)n1 C12(CNC(CCC(=C)Br)=O)CCC(CNC(=O)C(=O)N(C)C)(CC1)OC2 C1(CCCNC(c2ccc(C3CC3)cc2F)=O)CN(C(=O)C(F)C2CC2)CCO1 C1(NC(C(C)(C)SC)=O)CC(O)CN(C(=O)CCC(C)C)C1 CC1CC(NC(=O)CCC2CC2(Cl)Cl)CN(C(=O)COc2ccccc2)C1 c1(OC)cnc(Cl)[nH]c1=NC(=O)c1nc(-c2cc(C)c(F)c(C)c2)sc1C C1(NCCNC(c2ccc(CC)c(C)c2)c2nnnn2C)CC1C1CCCCC1 CC(C)C(O)Cc1cn(CCCNC(c2cn(C)nn2)=O)nn1 c1(OC)cc(C)cc(C(N2CCC3(CC2)CC3CNC(=O)CC(C)F)=O)c1O CC(C)CCC(C(=O)NCC1COCC(C)O1)NC(c1cn[nH]c1)=O N1(C(c2c(C)oc(Cl)n2)=O)CCOCC(C(=O)NC2C=CCCC2CO)C1 N1(C(C2(CNC(C3=C(C)CC3)=O)CCC2)=O)CCCCC(CN(C)C)C1 C1(CNC(CNC=O)=O)(CO)CC12CCN(C(c1coc(Br)c1)=O)CC2 c1(C(=O)NCC(CC)NC(c2c(C)nc(CCC)o2)=O)cncc(F)c1Cl c1(C(C)C)cc(C(N2CCC(C(C)NC(C3CC(=O)C3)=O)C2)=O)n[nH]1 C(CC1CC1)(CC(=O)NCCOC1CC1)NC(CCNC(COC)=O)=O CC1(C)CC=C(C(=O)N2C3CCC2CC(NC(=O)C2=CCCC2)C3)CC1 CC1CN(C(NC2CCCc3nc(O)ccc32)=O)c2cc(F)ccc2C(=O)N1 C=CCC(C)(C)CC(=O)NC1(C(=O)NC(C)C(F)(F)F)CCC1 C12(C(=O)NCCC3(NC(c4cc(CC5CCC5)c[nH]4)=O)CC3)CCCC1CC2 C1(CCOC)(NC(=O)CC(O)CN(C)C)CCN(C(=O)C(C)(C)C#N)CC1 N1(C(C(C)SCC)=O)CCCCCCC1C(=O)NCc1n[nH]cc1C c1(OC)ccc(-n2cccn2)cc1CNC(=NCC1CC1)NCC1(OC)CC1 C12(C(N3CC(C(C)(C)O)(CNC(CN(C)C)=O)C3)=O)CCCC1(C(N)=O)C2 C12CN(CCCO1)C(=O)N2.Cc1cc(-c2ccnc(CC(=O)O)c2)ccn1 N#Cc1nnc(N2CCC(=CCNC(c3ccc(C(F)F)cn3)=O)CC2)s1 C(C(C)(C(=O)NCC(C)(F)C(C)C)NC(=O)Cn1ncnn1)SC c1(NC(CC(C)NC(=O)CC(F)(F)C(F)F)C)ncnc2cnccc12 C1(NC(C2=CC(C)CC2)=O)CC2(CCN(C(C3CC3c3ccc(F)c(F)c3)=O)C2)C1 C1(N(C(=O)CS(=O)(=O)N(C)C)CC)CCC(NC(=O)CCc2cn(C)cn2)CC1 C(=O)(CCCCCC#N)NCC(C(C)(C)C)NC(c1c[nH]c2ccccc12)=O N1(C(C(N(C(=O)C=Cc2cc[nH]c2)C)C2CC2)=O)CC(C2(C)CC2)C1 C(C(=O)NC(C)(C)C(F)F)(C(C)C)NC(CC1C(CC)C1)=O Cc1cc(=NCC2CCN2C(C)(C)C)[nH]c(-c2cccnc2)n1 C(CC(C(=O)NC1CC(OCC)C1)NC(=O)C(C)N=[N+]=[N-])OCC C1(NC(C(C)(C)C(F)(F)F)=O)CC(C2CCN(C(c3cccc(O)c3F)=O)C2)C1 C1(CC(=O)NCCCCC(C)NC(c2c(C)scn2)=O)CC2(CCC2)CO1 CC1(C(=O)NCC2CC3CC2CN3C(=O)CCn2cnnn2)CCCCNC1=O c1(C(N2CCC(CNC(C3C(C(N)=O)C3)=O)C2)=O)nccnc1C(F)(F)F c1(Oc2c(NC(=O)NCC3C(=O)NC(=O)S3)cccc2)ccc(Cl)cc1Br C=CCC(C)(C)C(=O)NCCn1cc(C(=O)N(C2CCC2C)C)cn1 CC1(C(=O)NCCN(C(c2cc(Cl)c[nH]2)=O)Cc2ccccc2)CCC2CC2C1 Cc1cccc(C(N2C3CN(C(C4C=CCN4)=O)CC23)=O)c1[N+](=O)[O-] C1(C(N2CCC(C(N(C)C)=O)C2)=O)CCN(C(c2cccnc2O)=O)CC1 C1(C(=O)OC)CC(C(C)C)CCN1S(=O)(=O)CC(C#N)C1CCNCC1 n1(CC)cc(C(=O)N(CCC(N2CCC(C)(C(N)=O)C2)=O)C2CC2)c(C)n1 C1(NC(C(C)(C)OCC)=O)CN(C(C2CC2C)=O)CCC1c1ccc(F)cc1 N1(C(C(CCN(C)C)NC(CC(C)C)=O)=O)CCCCCCC1C C1(C(N(C)CC2(NC(c3ccc(CC)[nH]3)=O)CC2)=O)CC(F)(F)C1(C)C C1CCN=C2N=C(C=CN2)C(=O)O1.N1(C(=O)OC(C)(C)C)CC(=O)NC(=O)C1 N1(C(c2c(CC)nn[nH]2)=O)CC(F)(F)CC1CNC(=O)CCc1ncco1 CC(C)(CC(=O)N1CC(CNC(C2CC3(CCC3)CO2)=O)C(C)(C)C1)C(F)(F)F c1(C(=O)NC2(C(=O)NCC3(Cl)CCC3)CCSC2)cccnc1O C1(CNC(C2CC(CC)OCC2)=O)CCCCCN1C(c1cc2occc2[nH]1)=O N1(C(c2c(CNC(C3CC34CCC4)=O)cc[nH]2)=O)CC2(CC(O)C2)C1 C1(=CC(=O)NC(CNC(C(C)c2cc[nH]n2)=O)C2CCC2)CCC(C)(C)CC1 C1(CNC(C2C(C)CCC2)=O)CN(C(c2ccc(NC(C)C)cc2)=O)CCCO1 Cc1cc(F)ccc1NC(c1cc(C)c(Br)s1)c1nnnn1CCCC1CC1 Cn1cc(C(O)C(=O)NCC2CCCN2C(c2coc(O)n2)=O)cn1 N1(C(c2nc(C)sc2)=O)CCC2(CCN(C(=O)C(C)(C)C(C)(C)O)CC2)C(C)C1 C1(C(N(CC(C)O)CCNC(C2CN(C(=O)NC)C2)=O)=O)CCC(C(C)C)CC1 c1(N(CC=C)C)nnc(CCC2CCCO2)n1CC1CCCCO1 C(=O)(CCCc1nncn1C)N(C(C)C)CCNC(C1(n2cncn2)CC1)=O Cc1nc[nH]c1CC(=O)NCC(C)NC(=O)CNC(=O)NC1CC1 C1(C(=O)NC(C)(CNC(c2cnn(C3CC3)c2)=O)C2CCC2)CN(S(N)(=O)=O)C1 C(CCC(=O)NCCC1(C(=O)N(C2CCSC2)CC)CCC1)OCC c1(C(=O)NC2(C)CCN(C(=O)CCSCC(N)=O)CC2)ccc2c(n1)NCC2 C1(CC(=O)NCCOC2CCN(C(C3(C)ON=C(C)C3)=O)C2)CCCS(=O)(=O)C1 c1(C(N2C3CCC(NC(CCC=CC)=O)(C3)C2)=O)cccc2c1OCC2 Cc1cc(=O)c(C(N2CCC2CNC(=O)C(C)(O)C2CCC2)=O)cn1C N1(C(C=C(CC)C)=O)CCC2(CC1)CC2CNC(C1(CC(C)C)COC1)=O C(=O)(CC(C(C)(C)C)NC(=O)CC1CSCCO1)N1C(CC(N)=O)CCC1 C1(C(N2CCC(NC(c3ccc(C4CC4)s3)=O)C2)=O)OC2CCC1CC2 Cc1nc(C(=O)NC(C)(CNC(=O)COCc2cccnc2)C2CCC2)cs1 C1(CN(C)C(c2[nH]nnc2C2CC2)=O)COCCN1C(c1ncccc1Cl)=O C1(N(C(c2c(C)nsc2)=O)C)CCN(C(C2C3CCCCCCC23)=O)CC12CC2 N1(C(C(C(=O)OCC)F)=O)CCCC(C2(NC(c3oc(COC)cc3C)=O)CC2)C1 c1(N2CCC(CCNC(c3ccnn3CCF)=O)C2)cc(C(F)(F)F)nc(Cl)n1 c1(C(N2CCCC2Cn2cc(CC3CCCC3)nn2)=O)c(F)ccc2occc12 Cc1nc(N2CC(OCCNC(c3c(Cl)cnn3C)=O)C2)c(C)c(C)n1 C=CCC(C(=O)N(CC(O)CN(C)C(C1CC1C)=O)C)NC(C)=O c1(CN(C(C2N(C(CC3C(CC)C3)=O)CC(F)C2)=O)CC)cc(F)ccc1C C1(NC(C2CN(C)C2)=O)COC2(C1)CN(C(=O)Cc1cnns1)C2 C1(OC)CC2(CCC(C(N3CC(NC(c4nc5ccccc5o4)=O)C3)=O)CC2)C1 C1(C(N(C)CC2OCCN(C(CCCCN(C)C)=O)C2)=O)CC12CC(C)(C)C2 CC(C)CS(=O)(=O)CCC(=O)N1CCC(CF)(NC(=O)CC(O)C(C)C)C1 c1(C(C)C)nccn1CC(=O)NCCCN(C(=O)CC1OCCO1)C(C)C N1(CC(=O)N(C(C)=O)Cc2cccn2C)CC2CCC(C1)C2O c1(C(N(CCNC(C(C=C)C)=O)CC)=O)cnn2cccnc12 C(=O)(N1CCCc2ccnn21)c1c(CNC(C(CCCC)F)=O)noc1 Fc1ccc(I)c(CNC2CN(CC3CCC3)C2)c1 C1(NC(c2cccc(CC=C)c2)=O)CCN(C(C2(COCC)CC2)=O)CC1O CCCCC(O)C(=O)N1CC2CC2(NC(c2ccc(-c3cc(O)ns3)cc2)=O)C1 C(CCN(C)C)(C(=O)N1CCCC1CC1CC1)NC(c1nc(CC)sc1)=O c1(C(=O)NCCC2CCCN2C(c2ccc(Cl)s2)=O)ccnnc1Cl n1(CC(=O)NC(C2CN(C(c3c[nH]nc3F)=O)CCO2)C)cnc([N+](=O)[O-])n1 c1(C(N2CC3COCC3C2)=O)cnn2cc(-c3cc4c(F)cccc4[nH]3)ccc12 CC1(C)C(C(N2CCN(C(=O)CCc3nc(O)n[nH]3)CC23CC3)=O)CCS1(=O)=O c1(NCCCC(CC)O)ncnc(NCCN2CCC(C)(F)C2)c1C C1(COC)(CNC(c2cc3sccc3s2)=O)CCN(Cc2cc(C)no2)CC1 c1(C(=O)NC(C(CO)NC(CC)=O)C)cncc(C(=O)NC2CCC2)c1 C(=O)(C(C(C)CC)OC)N1C(CNC(c2nnn(CC)c2C)=O)C(C)CC1 N#CC1(C(N2CCOCC(NC(c3c[nH]cc3C(F)(F)F)=O)C2)=O)CC2CC2C1 C1(NC(CC(C)OCC)=O)CCC2(CCN(C(c3ccc(NC)cc3)=O)CC2)C1 C12(C(=O)NC(CC(=O)OCC)C)CC(CN(C(C3CCC(=O)CC3)=O)C1)C2 N1(C(c2c(C)n(C)nc2)=O)CCC2CCCN(C(=O)Cc3ccc(F)cn3)C2C1 OC12CCCC(CC(NCC3CC4CC(C3)C4)C1)C2 C12(CNC(C3CN(C4CCOC4)C3)=O)CCC(CC1)N(C(=O)C(F)C(F)(F)F)C2 C1(C(N2CC(C)C(NC(=O)CCCCCNC(N)=O)C2)=O)CC(=O)NC(=O)C1 CC1CCCCCC1NC(c1ccc(F)c(F)c1)=O CCCCCCCC(=O)NCC1CCC2(CCC2)C1NC(C1CS(=O)C1)=O c1(CN(C2CCCN(C(CC3C(C)CCO3)=O)C2)CCO)nnc2n1CCCCC2 c1(N2CCC(CN(CC(F)(F)F)CC)CC2)nc(=N)[nH]c(=NCC2CC=CC2)[nH]1 C1(C(N2CC=C(C)CC2)=O)CN(C(C2(C)CCCS2)=O)CC12CCC2 c1(C(N2CC(CC(=O)NC3(CC4CC4)CCOC3)(OC)C2)=O)c(F)cccc1F CC1(C)CCC=C(C(=O)NC2(CCNC(=O)Cn3cccn3)CCCC2)C1 O=C(C(O)CC(F)(F)F)NCC1C(C2CC2)CCN1C(c1cc(F)ccc1Cl)=O CCCCS(=O)(=O)NC(C(=O)N(CCC)CCNC(=O)C(O)C(C)C)C(C)C C#Cc1cccc(NC(C2CCCN2C(C2CCCC(F)C2)=O)=O)c1 C(C1=NOC2(CCC2)C1)N1CCC2C(CN)C2C1 C1(CCOC)CCN(C(=O)C=CCN(C)C(C2CC2C#N)=O)CC1 N1(C(c2nccc(C(=O)OC)c2)=O)CC2CCC1C(Nc1ncnc(Cl)c1F)C2 S(=O)(=O)(c1cccc(N2CCCc3[nH]ccc3C2)n1)N(CCCC=C)C c1(N(CC(=O)NCC(CNC(c2c(C)ocn2)=O)C)C)ccc(Cl)cc1C#N CCCC(C(=O)NCC1CN(C(C2CC(CF)C2)=O)CCO1)N(C)C C1(CC(N2CC(OC)C(NC(=O)C(F)(F)c3nccs3)C2)=O)CCC(F)(F)CO1 C1(CC(=O)NCc2c(C)nn(C)c2)C2CCCC2N1C(=O)CC1CCOC1 CC(C(F)C(=O)NCC1CCN(C(c2ccc([N+](=O)[O-])c(O)c2)=O)C1)C(F)(F)F c1(OC)cccc2sc(-c3nc(-c4ccsc4)nn3CCN(C)C)cc12 C1(C(=O)NC2CC(C(C)NC(COC(CC)CC)=O)C2)CCC(F)C1 N1(C(CCOCC(C)C)=O)CCN(C(C2CCC2)=O)CC1CC(F)F C(=O)(C1c2ccccc2CN1C(c1occc1C)=O)Nc1c(F)ccc(OC)c1 c1(C(=O)NCCC(CNC(C2CC3CCC(C2)C3)=O)OC)cn2ccccc2n1 C1(C(=O)NCc2cc(C(=O)NCC(C)(O)C3CCC3)n[nH]2)C2CCC(=O)C12 C=CC1CCCCN1C(=O)C(COC)NC(=O)CCCC1CCCO1 C1(C(N(C)Cc2nc(C)[nH]n2)=O)C2CCCC2CN1C(=O)C(Cl)Cl C1(CNC(CC2CC(C)C2)=O)CCCN(C(=O)Cn2nnc(-c3ccsc3)n2)C1 c1(N(C)C)cc(Br)ccc1C(N1CC=CC(NC(=O)CN2CCCC2=O)C1)=O c1(CC(C)C)cc(C(=O)NCC2CCN2C(C2CC2c2cccs2)=O)cc(O)n1 C1(C(=O)NC(CC)C(=O)NC)C=CCN(C(=O)C(C)c2ccco2)C1 C1(C)(CNC(c2nc(C(C)C)oc2)=O)CCCN1C(c1n[nH]c(C(C)(C)C)n1)=O N1(C(CNS(C)(=O)=O)=O)CCCOC(CNC(c2ncoc2C2CC2)=O)C1 Cc1sncc1C(=O)NCC(C1CCCCC1)NC(=O)CCn1cc(Cl)cn1 Cn1ncc(Br)c1C(N1CCC1CNC(C1(C(F)(F)F)CC=CC1)=O)=O C(=O)(CC(C)(C)C(F)F)N1C(CN(C(COCC#C)=O)CC)CCCC1 C=CCC(C)(CC)C(=O)NCC(C)CN(C)C(c1cnc(N)c(N)c1)=O N1(C(c2cc(C)[nH]n2)=O)CC2CC(NC(=O)CC3CC4(CC4)CO3)C1C2 C(=O)(CC(C(F)(F)F)OC)NCC(C1CCC1)NC(Cc1cc(CC)nn1C)=O c1(C2(C(=O)NC3C(NC(CN(C(=O)OC)C)=O)CCC3)CC2)ccc(F)c(Cl)c1 C1(CCC)CN(C(=O)Cc2ccco2)CCN1C(=O)CC1COCCN1C c1(NC2CCN(C(=O)OC(C)(C)C)C2C2CC2)cc(F)ccc1S(=O)(=O)CO C1(C(=O)NCc2ccc(OC)cn2)COCCN(C(c2ccno2)=O)C1 C1(SC)CCCC(NC(=NCc2ncccn2)NCc2ccnn2C)C1 c1(OC)ccc(C)c(OC)c1C(N1CC(NC(c2ncncc2Cl)=O)C1)=O N1(C(C(CCC)(C)C)=O)CCC2(CCC(CNC(=O)C(C)CC3CC3)OC2)CC1 c1(C(N2CCC(CNC(C3(C)C(C)C3)=O)C2)=O)c(N)cc(F)cc1Cl c1(-c2n(C(COC)C)nc(C3CC3)n2)ccc2c(c1)nnn2Cc1ccccc1 N1(Cc2cccc(OC)c2C)CCC(NC(=O)C(c2ccccc2)F)C(C)(C)C1 c1(SC)cc(C(=O)NCCC(C)N(C)C(c2sc(CO)nc2C)=O)c(C)o1 C1(NC(C(C#C)(C)C)=O)CC2CCCC(C1)N2C(=O)Cc1ccc(F)cc1F Cc1cnc(N)c(S(=O)(=O)N)c1.C1(C2(O)CCC2)(NCC(C)C(F)(F)F)CC1 Cc1cc(C(N2CCC(O)(C(N3CCCC3(C)CCCO)=O)C2)=O)c(C)n1C CCCCN=C(NCCC=C(C)C)NCC1CC1(Cl)Cl C=CC(CCC)CC(=O)NCC(CCC)C(=O)N(C1CCCCC1(C)O)C CC1CCc2nc(C(=O)NC3CNCCC3C#N)cn2C1 N1(C(C(C=C)O)=O)CCC(CNC(C2(CO)CC2(F)F)=O)(COC)CC1 C(=O)(C(C)CC(F)(F)F)NCCNC(c1c(C)nsc1N)=O C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NCCC(CCNC(C(CC)OC)=O)C Cc1cn(CC(N2CC(F)(C(=O)NCCC(=O)NC3CC3)C2)=O)c(=O)nc1O CC(O)C(C(=O)N1CCC(O)(CCNC(=O)CCc2ccccc2)C1)N(C)C c1(C(N2CC(CNC(C(CC)n3ccnc3)=O)C2)=O)cn2ccnc2cn1 C(C(C)(C)C(=O)N1CCC(C(F)C(=O)Nc2ccc(N(C)C)cc2)C1)OC C1(C#N)(NC(C2(C)CCCC2)=O)CCN(Cc2ccc(O)cc2)C1 c1(C(N(CCN(C(c2c(C)nccn2)=O)C)C)=O)ccc2ccnc(O)c2n1 c1(C(=O)NC2C(NC(CC(C)C3CC3)=O)C2)cnc(=N)[nH]c1 c1(CC)c(C(N2CC3CC3(C(=O)NC3CC3c3ccc(F)nc3)C2)=O)cnn1C C1(CCOC)(NC(=O)C(c2ccc(C)cc2)C)CCN(C(=O)CNS(N)(=O)=O)C1 c1(C(=O)NC2CN(C(C(CCSC)NC(N)=O)=O)CC2O)cnc2sccn12 C1(C(N2CC(COC)(CNC(c3cc(Cl)cnn3)=O)C2)=O)OCCOC12CCC2 C1(CNC(C2CCC(O)C2)=O)CC2CCC1N(C(c1cncc(Br)c1)=O)C2 c1(CCC)cc(NC(=O)C(C)(c2ccccc2)NC(=O)NC)c(C)o1 CC1CN(Cc2ccccc2)CCN1N1CCC(F)(F)C(C)C1 c1(C(C)(C(=O)O)OC(C)=O)cccc(Cl)c1.N1(C(CC2(CC(=O)OC)CC2)=O)CCCC1 Cc1[nH]nc(O)c1NC(=O)NC1(C)CC1(C)C N1(C(CC2C(C)(C)OCCO2)=O)CCN(C(c2cccc(N)c2F)=O)CC(O)C1 Cc1cc(C(N2CCC(F)(C(N3CCOC(CCF)C3)=O)CC2)=O)cc(C)n1 C(=O)(C(C(C)CCCC)N1CCCC(OCC)C1)NCC=C.C(C)(C)(C)ON Cc1ccc(C=CC(=O)NCC(C(C)C(C)C)NC(c2cnc(O)o2)=O)cc1Cl c1(NC(N2CCN(C(C(=O)NC)C)CC2)=O)cc(F)cnc1CO CCC(C#N)C(=O)N(O)Cc1cn(C(C)C(=O)Nc2nn(C)cc2C)nn1 C1(NC(C(C)OC2CCCCC2)=O)CCN(C(c2cnnn2C2CC2)=O)CC1C N1(C(CCCCC)=O)CC(O)(C2(CNC(=O)C(CC)C(=O)OC)CC2)C1 C(=O)(C1CCc2c[nH]nc21)N1C(CNC(CCc2c(C)noc2Cl)=O)CC(F)C1 C1(CNC(Cc2cn(C)nn2)=O)(CO)CCN(C(=O)CCCc2cc[nH]n2)CC1 C1(C(N2CCC(NC(=O)CCc3ccoc3)C2)=O)CCCc2ccccc2C1 C1(C(=O)NCC(CC)N(C(=O)Cc2cccc(C)c2)C)CCN(OC)CC1 c1(SC)ccc(-c2csc(C(N3CCC(C)(C)CC3)=O)n2)c(C(F)(F)F)c1 C=CCC(CNC(c1cc(C2CC2)[nH]n1)=O)C(=O)N1CCCC(F)CC1 N1(C(c2c(F)ccc(N)c2F)=O)C2CCC1C(F)C(NC(C1CCSC1)=O)C2 CC1(C(=O)NCC2(CNC(C3CCCCC3(F)F)=O)CC2)CCCCCC1 c1(NC(C(CC)C)c2nnnn2-c2cccs2)ccc(-n2cccc2)c(Cl)c1 N1(C(c2cc(C(C)=O)[nH]n2)=O)CCCC1(C)C(=O)NC(c1cccc(C)c1)CO c1(C(=O)OCCC23CC(CCO2)C3)n[nH]c2ccc(C(F)(F)F)cc12 Cc1ccc(CC(=O)NC(C)(C)CCCNC(=O)CCCCC#N)cc1O N1(C(c2occ(C)c2)=O)CC(O)(C2CCN(C(C3CC4CCC4C3)=O)CC2)C1 Cc1cc(C(=O)NCC2CCCC2NC(=O)CC2COC(=O)C2)cc(O)n1 c1(C(=O)NC2C(CNC(Cn3ccc(C)n3)=O)CCC2)c(C)nn2c1NCCC2 C1(F)(CNC(c2n(CC)nnc2C)=O)CCCN(C(=O)CCS(N)(=O)=O)C1 CC12CC(NC(=O)NCC3(CC4CC4)CCOC3)(C1)C2 c1(CCC(C)NCCCc2ccc(Br)cc2)ccc(C(F)(F)F)cc1 C(CCF)(C(=O)NCC1(O)CCC(C)C1)NC(C1C=C(C)CS1)=O C(=O)(CCCC(=O)N1CC(NC(c2c(C)noc2CCC)=O)CC1C)NCCC Cc1ccc(C(=O)NC(Cc2ccoc2)C(=O)NCCc2c[nH]nc2O)c(F)c1 CC1CC(NC(=O)Cc2nc[nH]n2)CN(C(c2nnc(O)cc2O)=O)C1 C1(NC(c2ccc(CC)o2)=O)CCN(C(=O)C(O)C(F)F)C1c1ccccc1 c1(C(=O)NC2C(C(=O)Nc3c(C(=O)OC)onc3C)C2)c(C)cccc1Br C(C1=CCN(C(C2CCCC(=O)O2)=O)CC1)NC(CC=C(C)C)=O CC1CCc2cc(C#N)c(N3CC(C)(NC(c4cc(Br)co4)=O)C3)nc2C1 c1(C(N2CCC3(CCN(C(C(C)OCC)=O)C3)C2)=O)ccc2c(c1)C=CS2(=O)=O N1(C(C(C)N(C(=O)CCc2nc(O)n[nH]2)CC)=O)CCOC(C)(C)C1C C1(CC(=O)NC2(CN(C(c3c(OC)nsc3)=O)C)CC2)CCC(=O)NC1 CCC(C(=O)NCCC1CCCN1C(c1cnsn1)=O)NC(C)=O c1(CC)c(NC(C2CN(C(=O)C(C)(Cl)Cl)CC2C)=O)cnn1CC N1(CC(=O)NCCCN(C(c2cnc(-c3ccco3)s2)=O)CC)C(=O)CNC1=O N1(C(C2N(C(C)=O)CC(O)C2)=O)CCCC(N(c2ncc(Br)cn2)CCO)CC1 C1(NC(c2conc2C2CCCC2)=O)Cc2cscc2C1 c1(NC(=O)Cc2cc(C3(C4CCCC4)CC3)on2)ccccc1Br c1(-c2n(CC)nc(-c3ccc(CN(C)CC)cc3)n2)cc2cc(F)c(F)cc2[nH]1 c1(C(=O)NCC2C(NC(CC(C)CN(C)C)=O)C2)ccc2cc(F)ccc2n1 C(=O)(C(O)CC(C)(C)C)NC1CC(O)(CNC(c2c(C)n[nH]c2C)=O)C1 c1(C(=O)NC(CNC(=O)C=CCn2cncn2)C2CC2)cc(F)cc2c1NCCC2 N1(C(C(C2CCC2)OC)=O)CCC(C2CC2)(NC(c2ccns2)=O)C1 c1(C(=O)NCC2C(NC(c3cnc(O)s3)=O)C2)ncccc1N1CCOCC1 C1(NC(c2c(CC)occ2)=O)CCN(C(=O)CSCC(=O)OC(C)(C)C)C(C)C1 N1(C(CCOCC(C)C)=O)CCC(NC(=O)C=CC2CCOC2)C(C)(C)C1 c1(C(=O)NC2CCC(NC(c3c(C)ccc(C(N)=O)c3)=O)C2)cc2c(cn1)OCO2 Cc1ccc(C(N2CC(NC(c3c(O)cccc3F)=O)CC(C)C2)=O)c(F)c1F n1(CC)nc(C(=O)NCC(C)(C)CNC(C23CCC(CC2)O3)=O)cc1C(F)(F)F N1(C(c2cc3c(s2)CCOC3)C(=O)NCc2ccco2)Cc2ccc(O)cc2C1 C1(NC(C(CC)C)=O)C=CCN(C(c2cc(-c3ccc(Cl)cc3)no2)=O)C1 C=CCC(C(=O)NCC1CC(C)(C)CN1C(c1ccn(C)n1)=O)C(C)C C1(C(=O)NCc2cc(C)ncc2)CN(C(c2cc(Cl)cs2)=O)C(C)(C)C1 C1(NC(CCC(=O)NC)=O)CN(C(c2cc(N)c(F)cn2)=O)C2(CCOCC2)C1 N1(CCNC(C2CCCOCC2)=O)CCN(C(c2cnc(O)o2)=O)CC12CCC2 Cc1cc2ncc(C(=O)NCC3CCN3C(=O)CC3CC4CC4C3)c(C)n2n1 CC1=NOC(C)(C(=O)NC(C)CNC(=O)CC2(C)CC2(Cl)Cl)C1 C(=O)(CN=c1[nH]c(C)cs1)NCCOC1CCN(C(C2CC3(CC(=C)C3)C2)=O)C1 C1(C)(C(N2CC(CC3CC3)C2)=O)CCC(C(=O)NCC2(CC)CCC2)O1 C1(C(=O)NCC(C(=O)NCC)(C)C)CC2(C1)CN(C(C1CN(C(C)=O)C1)=O)C2 c1(C(=O)NCC(C2CC2)Nc2ccc(C(=O)OC)cn2)cnc2cc(C)nn2c1 C(C(CC(F)(F)F)NC(C1CCCOC1c1ncc[nH]1)=O)NC(C=C(COC)C)=O Cc1c(C(=O)NC2(C)CCN(C(=O)CCC(C)O)CC2)oc2c(F)cccc12 c1(C(N(CCN(C(C2C(C(C)C)OCC2)=O)C)C)=O)cn2ccnc2cn1 c1(C(C(=O)NC(CC)(C)C)N(C2CCCCC2(C)C)C)n[nH]c2c(Cl)cccc12 Cc1cn2cc(C(=O)NCC3(C)CC(F)(F)CN3c3ccnc(C)n3)sc2n1 C1(NC(=O)CNC(=O)C2CC2)CCOCC1NC(c1cn(C2CCC2)nn1)=O c1(C(=O)NC(C)CC2CN(C(=O)CCCC#N)C2)ccn2c1CS(=O)(=O)CC2 N1(C(CC=CCCCCC)=O)CCN(C(c2cc(C)sc2N)=O)CC1 N1(C(c2ccc(C3(C#N)CC3)cc2)=O)CCOCC(CNC(C2CC2CF)=O)C1 c1(C(=O)NCC2(F)CC(NC(CCC#C)=O)C2)ccccc1CS(C)(=O)=O N1(C(C2C(C)C2)=O)CCC2CCC(NC(=O)C=Cc3ccn(C)c3)C12 CN1CCN(C(C2CC3COCC3C2)=O)C(CNC(c2n[nH]cc2[N+](=O)[O-])=O)C1 n1(CCC2(C)CC2)cc(C#CC(C)(C)NC(=O)Cc2cccc(Br)c2)nn1 c1(C(=O)NCC2N(C(COCCC)=O)CCC2C2CC2)cc(F)c2c(c1)CCC2 CCCC(O)CC(=O)NCC1CCN(Cc2cc(C3CCCCC3)on2)C1 c1(C(N2CCC(CNC(C#CC)=O)CC2)=O)ccc(=O)n(C(C)C)c1 CC(C)CC(C)(O)C(=O)N1CC2=C(C1)CN(C(=O)C(C)Cc1cnco1)C2 CCC(C)(C)C(=O)NCC1(F)CC(NC(C2CC(CC(F)F)C2)=O)C1 CCCCC(CC)N=c1[nH]c(=NC)[nH]c(=NCCCc2[nH][nH]c(=N)c2C#N)[nH]1 CCCCCC(O)C(=O)N1CC(NC(c2nnc(C)cc2O)=O)CC(C)(C)C1 C1(C(C(=O)OC)(C)C)CCCN(C(c2c(C)noc2C)C(=O)NC(C)(C)C)C1 Cc1oc(C(C)(C)C)cc1C(=O)NCC1CCCN1C(N)=O N1(C(c2ncccc2Cl)=O)CCCC(C2CC2NC(C2CC(CC3CC3)C2)=O)C1 C1(CNC(C)=O)CCC(NC(C2CCOC(C)C2)=O)CC1 C1(NC(C2N(C(CC3(OCC)CCC3)=O)CC(O)C2)=O)CCC2(CCC2)C1 Cn1cc(C(N2CC3CC3C2C(N2CCCC(C(N)=O)C2)=O)=O)ncc1=O c1(OC(CC)C)ccccc1NC(N1CCN(CCOC)CC1)=O c1(C(=O)NC2(COC)CN(C(C3C=CCC3)=O)C2)[nH]c2ccc(F)cc2c1C C(=O)(C(O)CC(C)(C)C)NC(CCCC)CNC(c1ccc(C(C)C)c(F)c1)=O C(c1ccc(F)c2ccccc12)=CC(=O)NC1CC(c2ccc(F)cc2)(CO)C1 c1(OCC(=O)NCC(C)(C)Nc2nc(-c3cccnc3)cs2)ccc(F)cc1 C(=O)(CC(C(=O)NC1CN(C(=O)C(C(C)C)SC)C1)N1CCCCC1)OC CC1CCC=C1C(=O)NCCC1CC(NC(c2ccc(SC3CC3)cc2)=O)C1 N(C1COc2cc(Br)cc(F)c21)C(N1CCCC(F)(CO)C1)=O c1(C(=O)Nc2nc(Cl)ccc2I)ccc2c(C(=O)N=c3cco[nH]3)n[nH]c2c1 N1(C(c2cnc(Cl)[nH]2)=O)CCCC2(CCN(C(=O)C3COc4ccccc43)C2)C1 C1(NC(C2(C)CC=CCC2)=O)CC2(CCCCN2C(=O)CCC2CC2(F)F)C1 C(C(C(=O)NC(C)C(=O)NCC(C)C)C(C)C)NC(c1n(CC)nnc1)=O C=CC(CCC)CC(=O)NC1CCCCC1NC(c1cnn2ncccc12)=O C=CCC(CNC(c1ccc(C2CC2)o1)=O)C(=O)NC1C=C(C)CCC1 CC1=C(C(=O)NC2CCN(C(C3(CN(C)C)CC3)=O)CC2F)CCO1 c1(SC)cc(C(=O)N(CCCNC(=O)CC2C=CCCC2)CCO)oc1C n1(CC(=O)NC(CN2CCN(C(CCOCC)=O)CC2)(C)C)cc(F)ccc1=O c1(C(N(CCOCCNC(c2n[nH]c(C)c2O)=O)C)=O)cc2cscc2s1 c1(C(N2CC(N(C(=O)CCC3CCCN3C)C)C2)=O)coc2c1C(O)CCC2 c1(C(C(=O)Nc2cccs2)NC(C(CCC)NC(C)(C)C)=O)ccc(Cl)cc1Cl c1(C(C)OC(=O)COCCC2CC2(Cl)Cl)ccc2c(c1)CCC2 C1(CCOC)CN(C(c2ncn(C(C)(C)C)n2)=O)CCN1C(=O)CCCN=[N+]=[N-] C1(C(=O)NCCC(=C)CSC)CC2CCC(C1)N2C(=O)C(C)Cc1cnc[nH]1 Cc1nn(CC(N2CC(CNC(C3CC3CF)=O)C(O)C2)=O)cc1Br c1(C(=O)NC(C2(C(N(CCSC)CC)=O)CC2)C)ccc(C)c(F)c1 C1(NC(CCCN(C(=O)OC)C)=O)(CO)CCN(C(C2CCSC2)=O)CC1 c1(CNC(C(C=CC)O)=O)cc(C(=O)NCc2nnnn2CCC)ncn1 c1(C(=O)NC2CCN(C(C=COC)=O)CCC2CO)cnc(O)c2ccccc12 C1(C(=O)NCC(CCNC(C2(CC)CCCO2)=O)O)CC(=O)N(O)C1 C1(C(=O)NCCN(C(Cc2c(C)noc2Cl)=O)C)CCc2cn(C)nc2C1 N1(C(C(C)NC(c2ccc(NC)cc2)=O)=O)CC2CCN(C(=O)CC(C)(F)F)C2C1 C1(C(=O)NCC2N(C(C(C)C3CCC3)=O)CC2)CC2CC1C1C2C1(F)F c1(N(CC(C)CNC(=O)C(C)(C)C)C)nccc(CO)n1 c1(C(N2CC3C(NC(CCc4ccc(CC)cc4)=O)C3C2)=O)ccc(Cl)c(O)c1 C(=O)(CCC1=CCCCC1)NC1CCN(C(C(CCC)OCC)=O)C1 Cc1ccc(C=CC(=O)NC(C)CC2CN(C(=O)CC(F)F)C2)s1 N1(C(c2n(C)cc(C#N)c2)=O)CCC(C2CC2NC(=O)C(O)c2ccsc2)CC1 N1(C(CCC=C=C)=O)CCN(C(C2CC2C2CCCC2)=O)CC2(C)CCCC12 c1(C(C(=O)NCC(=C)C)N(CC(C)(C)COC)C)ccc(C(F)F)cc1Cl c1(C(C)NC(=O)C=CCC(C)(C)NC(=O)CC2CC2(C)C)nn(C)cc1O C(=O)(C#CC(C)(C)O)N1C(C(N(CC(CC)(O)CC)C2CC2)=O)CC(O)C1 c1(CC)c[nH]cc1C(=O)N(CCNC(=O)Cc1csc(C2CCCC2)n1)CC Cc1ccc(C(N2CC3CC2CN(C(c2cn(C)nc2O)=O)C3)=O)c(N)c1F CCC(CCC(=O)NC(C)CCF)NC(c1ccc(C(C)=O)o1)=O C1(C(N2C(C3CCN(C(c4ocnc4C4CC4)=O)C3)CCC2)=O)CCS(=O)(=O)CC1 CCCCC(CNC(=O)CCCOCCC)NC(c1nccn1CC)=O NS(=O)(=O)c1cnn(CC(N2CCCC2CNC(c2cccs2)=O)=O)c1 c1(C(=O)NCC2CCN(Cc3onc(C(C)C)n3)C2)cnn2ccn(C)c12 c1(C(=O)NCCN(C2CCCCC2)C(C2CC23CC3)=O)cnc(C(F)(F)F)cn1 N1(C(CCC2CC(OC)C2)=O)CCC(CNC(=O)CC2CSCCO2)C1(C)C C(=O)(CC(F)(F)C(F)F)NCC12CCN(CC1)CC2.CC12CCN(C1)C(=O)C2 c1(OC)cccc(C(=O)N(CCCCCCNC(C2CCCS2(=O)=O)=O)C)c1 n1(CCC(=O)NCCCSCCO)c(=O)oc2ccccc12 C1(c2ccccn2)CCCN(CC(=O)N)C1.C(C)(CNC(C)=O)N(CCOCC)CC c12ccc(F)c(c1)C2.c1(CNc2cccnc2)ncsc1Br.O=C1C(C2CC2)N1 n1(CC)ncnc1C(=O)NCCOC1CN(C(=O)CC2(COC)CC2)C1 c1(C(=O)NC(CC)CNC(=O)C(C)n2ccnn2)oc(P(C)(C)=O)cc1C c1(C(N2CC(OCCNC(C(C)NC3CC3)=O)C2)=O)cnnn1C1CCCCC1 c1(C(N(CCC(=O)NC(COC)C2CC2)C2CCC2)=O)cccc(O)n1 CCC(O)CCCN=C(NCCOC(C)C)NC1CCC(=O)NC1 N1(C(C#CC(C)C)=O)CCC2(CCCC2NC(c2cc(O)cc(F)c2)=O)C1 N1(C(=O)CN2CCOCC2)CCN(C(C2CCCC3CC23)=O)CC1 c1(CNC(C2CCC(C)N2C(=O)COc2ccsn2)=O)ccnc(F)c1F c1(C(N2CC(CNC(C3CC4(CCC4)C3)=O)OCC2)=O)ccc2ncsc2c1 Cc1cccc2cc(NC(C3CC4CC3CN4C(c3n[nH]c(=N)[nH]3)=O)=O)sc12 C1(C(=O)NC(c2cccc(Cl)c2)c2cccc(Cl)c2)CCS(=O)(=O)C1 C(=O)(C(C1CCC1)N(C(=O)CCn1cnnn1)C(C)=O)N(CCCC)CCCO N1(C(c2nc(CC)oc2)=O)CC2CC(NC(c3cn(C4CC4)nn3)=O)CC2C1 C(CCO)(C(F)F)N(C(=O)NC(c1cccnc1)C)C Cc1ccc2c(N3C(CC)C(C(C)C)C3)ncnc2c1 c1(CNC(C2(OC)CCC2)=O)ccccc1CNC(c1n[nH]c(C)n1)=O c1(C(C)(C)C)cccc(C(=O)NCC2C=CC(NC(C3CCCN3N=O)=O)C2)n1 N1(C(C(c2c(C)cccc2)(F)F)=O)CC(NC(c2sccc2F)=O)C2CC2C1 c1(CN=C(NC2(C)CN(CC)C2)NCC2CC2)ccc2c(c1)n(C)c(=O)n2C c1(NC(CCCC)C)ccc(S(=O)(=O)N(C2CC=CCC2)C)cn1 C#CCC(CC#C)C(=O)NCC(CC=C)NC(=O)COc1ccc(F)cc1F C1(O)(CNC(c2c(C)cncc2)=O)CCCN(C(C2CC23CC(C)(C)C3)=O)CC1 CC(CN=c1ccc2ncc[nH]c-2n1)N(C)C(C1CCc2ncncc2C1)=O C1(C)(CCNC(C2(OC)CC(C)C2)=O)CCN(C(=O)C(C)(C)c2ccno2)C1 N1(C(CC(CC=C)(C)C)=O)CCCC2CN(C(=O)C=CCOC)CCCC12 C#CCC(C)(C(=O)NCc1cc(F)ccc1C)NC(=O)C=CCOC C1(NC(CC2C(=O)NC(=N)S2)=O)COC2(C1)CN(C(C1CCS(=O)(=O)N1)=O)C2 C#CCCC(C(=O)NC1CCC(O)CC1)NC(=O)CC1C(C)(C)C1(C)C N1(C(c2c(C)snn2)=O)CCC(CCNC(c2ccsc2C#N)=O)CC1C Cc1ncccc1C(N1CC(NC(=O)C(c2cccnc2)C)C1)=O C1(C(=O)NC(CCC)C2CCC2)CCCN(C(=O)CNC(=O)OC)CC1 C(CCC(=O)NC(C)CCNC(C1(C(C)(C)C)CCCC1)=O)OC(C)C C1(CNC(CCOC(C)=O)=O)CN(C(=O)COc2ccc(C#N)cc2)CCC1C N1(C(C(c2cccs2)SC)=O)CCN(C(C2(C)CCCCC2)=O)C2(CC2)C1 C1(NC(c2cn(-c3ncccn3)cn2)=O)CCN(C(=O)Cc2ccc(Cl)s2)C1 c1(CCC)cc(C(=O)NC(C)(C)CNC(=O)Cc2ccc(Cl)cn2)ccn1 CN1CCn2nc(C(=O)NCC(F)CNC(C3(n4cccn4)CC3)=O)cc2C1 c1(C(N2CCC(NC(C3CN(C)C(=O)C3)=O)C(F)C2)=O)nnc2n1CCCC2 N1(C(c2c(C(C)C)cnn2C)=O)CCC(NC(=O)Cc2ccsn2)CC(C)(C)C1 CC(C)C(C)(C)C(=O)NCCN(C(=O)C=Cc1cn[nH]c1)C c1(C(=O)NCC(CNC(C2(C(C)C)CC2)=O)F)ccc2occc2c1 C1(C(N2C(CNC(CC3(C)CC3)=O)CC3(CC3)C2)=O)CC2CCCC(C1)C2 N1(C(C(C)OCCN(C)C)=O)CCOC(CCNC(C2CCC3CC23)=O)C1 c1(C(=O)NC2CN(C(CCCC(CC)(C)C)=O)CC2C)cc2ccc(Cl)cc2s1 C(=O)(CCCC(F)(F)CO)N1CC2(C(NC(c3nn(C)c(O)c3)=O)CC2)C1 C(=O)(C(O)C(F)(F)F)NC(C1CC=CCC1)C(=O)N(CCC(C)O)C CC(C)CC(CN=c1[nH]c2ccc(Cl)cc2s1)NC(=O)CCN1CCCCCC1 C(C(C)(C)C(=O)NCC12CC(NC(C3CC(N4CCCC4)C3)=O)(C1)C2)SC.NC Cc1c(C(N2CCC(NC(c3cccc(F)c3)=O)C(F)C2)=O)ccc2c1CCC2 c1(C(N2CC3C(CNC(C4ON=C(CC)C4)=O)C3C2)=O)cc2c(cn1)CCCC2 C1C(CC(F)(F)F)NC(=O)N1.C1(C2CC2)(COC(C(C)C)=O)CCCO1.C(C)(C)(C)O Cc1cccc(C(N2CC(CCCCNC(=O)C(C)CN(C)C)C2)=O)c1C#N C1(CNC(CC=CCCCCC)=O)CCCN(C2CCN(CC(F)(F)F)C2=O)C1 C#Cc1ccc(F)c(C(=O)NC2CN(C(C3(C(N)=O)CC3)=O)CC2O)c1 C=CC(CC)CC(=O)NC1(CCOC)CCN(C(C2CCN(C)C2C)=O)CC1 C12CCCCC1n1cc(nn1)C2.CC1(C(=O)Nn2ccsc2=O)CC1(F)F N1(C(C(C#C)(C)C)=O)CCCC2(CCC(NC(c3ccc(Cl)cc3)=O)C2)C1 c12cc(ccc1O)CN2.n1(CC)ccnc1C1OCCC1NC(=O)OC(C)(C)C CCCCC(CC)C(=O)NC(CNC(=O)C=CCOC)C1CCC1 c1(CC(=O)NCC2CCCN(C(=O)CCc3nccs3)C2)coc2ccccc12 CCCCC(CC(=O)NC1CCC(=O)NC1)NC(=O)Cn1ccc(C)c1 c1(SC)ccc(C=CC(N2CC(NC(=O)CC(C)(C)C)CC(F)C2)=O)cc1 C1(OC)CCN(C(C2C3CCCC3CN2C(c2cc(C)nn2C)=O)=O)CC1(C)C CC1CN(C)CC1NC(c1c(CNC(=O)CCCCC2CC2)cnn1C)=O c1(C(N2CCC(C)(CNC(c3n(CC)ncn3)=O)C2)=O)cc(C(C)C)nc(O)c1 CC(C)(CC(=O)NCC1(C2CC2)CCN(C(C2(F)CCC2)=O)C1)C(F)(F)F C1(NC(CC2N(C)CC=CC2)=O)CC=C(C(=O)NCCn2cccn2)C1 C1(C(N2CC(O)(CCNC(=O)C(F)n3ccnc3)C2)=O)CC2C(C1)C2(F)F c1(OC)ccc(CS(C)(=O)=O)cc1C(N1CCCC(C(C)O)C1)=O CCC(CC(C)C)C(=O)NC1(C2CN(C(c3cc(C)n(C4CC4)c3C)=O)C2)CC1 C=C(C)CC(C(=O)OCC)NC(=O)CN1CCN(C(C2CCCO2)=O)CC1 N1(C(C2C(C)C2)=O)CCC(C2CCN(C(c3ccc([N+](=O)[O-])n3C)=O)C2)CC1 CCC(C(=O)N1CCC(NC(=O)Cc2c(C)n[nH]c2C)C(C(N)=O)C1)C(C)(F)F C(CC(C(=O)N1CCC1CC(=O)OC)NC(=O)C1=NOCC1)OC c1(C(=O)OC)ccc2nc(NC(CC3CCOC3)CO)cn2c1 c1(C(=O)NC2CCCC(N(C(CSCC#C)=O)C)C2)c(C)cc(OC)cc1F C=CC(C)(CCOC)C(=O)N(C(CNC(=O)CCCCO)Cc1ccccc1)C C1(CC(=O)NCC2N(C(Cc3scc(C)c3)=O)CCCC2)CCn2cncc2C1 C(C(F)C(=O)NC1(C)CN(C(N)=O)C1)C1CN(C(C(N2CCCCC2)C)=O)C1 N1(C(CC(CCC)(C)C)=O)CCN(C(C2CC2(C)C)=O)C2CCCC12 c1(NCc2ncc(C)c(OCC)c2C)ncc2c(n1)CCC(C(=O)O)C2 C(=O)(C1COc2ccccc21)NCCN(C(c1ncoc1C1CC1)=O)C1CC1 C#CCC(C(=O)NCCC(O)CCO)NC(c1cnncc1O)=O N1(C(=O)Cc2cc(C(=O)O)cs2)CC(F)CC1C(=O)NC(C)CC1(O)CCC1 C12CCN(CC1)C2.c1ccc(Cc2noc(C3CCCC3)n2)cc1 N1(C(N)=O)CCCC(C(N2CCOCC2c2cccs2)=O)C1 c1(-c2nc(C(CC)C)nn2C(C)C(C)C)ccc(Cl)cc1OC C1(C(NC(C(=O)Nc2scc(C3(C#N)CC3)n2)=O)C2CC2)CC2(CCNCC2)C(=O)O1 CCC1=NOC(CC(=O)NC2CC23CC(CNC(=O)CC(Cl)Cl)C3)C1 Cc1cc(C(=O)NC(C2CN(C(C3CC(CF)C3)=O)C2)C)cc(C)c1 N1(C(CC(C)(C2CCC2)N(C)C)=O)CCC(NC(c2cc(=O)n(C)o2)=O)C(O)C1 c1(C(N2CC3C(N(C(C=CC(C)C)=O)C)C3C2)=O)cccc(F)c1C#N c1(C(c2nnnn2C2CCOC2)NCC(CC)CC(C)C)cc2ccccc2o1 c1(OC)cc(Br)c(CNCc2ccsc2Cl)cc1OC C(=O)(C(N)C[Si](C)(C)C)NC(C1CCN(C(C)C)C1)=O c1(C(N2CCC(F)(c3cn(CCS(CC)(=O)=O)nn3)C2)=O)csc2nccn12 C(=O)(C1CCc2ccc(OC)cc21)NCC1(NC(C(CC=CC)C)=O)CCCC1 S(=O)(=O)(c1ccc(=NCCOC)[nH]c1)N(CCOC)CC1(F)CC(NC(C)=O)C1 C(c1ccc(F)cc1)=CC(N1CCCC1CCC(=O)Nc1ncn(C)c1)=O N1(c2c(C(=O)OC)cc(C)cn2)CCC(F)(F)C(NC(=O)CCCC2CCC2)C1 c1(CCNC(=O)NC(C)(C)CNC(=O)OC(C)(C)C)c(F)cc(Cl)cc1F Cc1cc2cc(C(=O)NC3CCCN(C(C4CC5(CC5)CO4)=O)C3)ccc2cn1 Cc1nc(C2CCCOC2)sc1C(=O)NCC1CC2CC2N1C(=O)CC1CCC1 Cc1ccc(NCC2CCC(NC(c3cnn(CC(C)C)c3)=O)C2)c([N+](=O)[O-])c1 c1(OC(CN(CCC)CCC#N)=O)cc(OC)cc(C(F)(F)F)c1 N1(C(CN(CCCCCC)C)=O)CCCCC1C(=O)Nc1ccccc1C c1(C(C(=O)NCCC(C)NC(C(CSC)C)=O)(F)F)cccc(Br)n1 C(COC(C)C)(C(=O)NC(CNC(C12CC(CO1)C2)=O)CO)NC(C)=O c1(C(=O)NCC2(NC(C(C)OCCC#C)=O)CCCC2)cc(Cl)c2n[nH]cc2c1 C1(C2C(NC(CCC=C)=O)CCO2)CCN(C(C2CC2c2cnn(C)c2)=O)CC1 c1(C(N2CC(CO)CC(OCCOC)C2)=O)ccc2cc[nH]c2c1F c1(C2C(C(N3CCC(F)(CNC(C(CCC)C)=O)C3)=O)C2)ccc(C#N)cc1 c1(C(=O)NC2CN(C(CN(C)CC)=O)CC2F)cc2cc(Cl)ccc2[nH]1 c1(C(N(C(CNC(=O)C(O)Cc2cnc[nH]2)C2CC2)C)=O)nc[nH]c2nccc1-2 CS(=O)(=NCC(=O)NCCSCCC(F)(F)F)c1ccc(Cl)cc1 C1(CN(CC(c2nnnn2C2CCC2)(C)NC(=O)OC(C)(C)C)C)CC(C)(C)CCO1 N1(C(=O)CSCC2CCCO2)CC2(CCC2)CC1CNC(C1CCC=CCC1)=O C1(C(N2CCC(C(C)NC(CCCOCC)=O)CC2)=O)CC2(CCC2)CO1 c1(NC(c2cc(CC)n(CCO)n2)=O)ccc(Cl)c(-c2cn(CCCO)nn2)c1 C1(CNC(C(C)NC=O)=O)CN(C(=O)Cc2cnnn2C)CC1N(C)C C(CCC(C)NC(=O)C(C)C#N)NC(C1(SCC)CC1)=O CN1N=C(CC(=O)NC2(CNC(C3CCCN3C(=O)C(F)(F)F)=O)CC2)CC1=O C1(CN(C(COCCC=C)=O)CC)CCCCN1C(=O)CN(c1ccncc1)C c1(CC)ccc(F)c(C(=O)NCCCCCNC(C2CCCC(O)C2)=O)c1F C1(C(=O)NCC2(CNC(CNS(NC)(=O)=O)=O)CC23CCC3)COCCN1C=O C(=O)(C1=CCC(C)(C)CC1)NCC(C)=CC(=O)NC(C1CCCO1)C1CC1 CC1(C)CC(C(=O)NCC(CC(F)(F)F)NC(c2ncccn2)=O)CC(C)(C)C1 N1(C(c2cc(C)ns2)=O)CCC2CC(C1)CN(C(C1CC1C1CC1)=O)C2 CC1(NC(=O)CN2CC3CC3C2)CCN(C(c2ncncc2Cl)=O)C1 C(=O)(C1=NOCC1)NC1CCC(NC(c2c(OCC)scc2)=O)C1 CCCCCCC(=O)NC1CN(C(=O)C(C)NC(=O)Nc2cc(C)ccc2Cl)C1 C1(NC(C2(C)CCCCC2)=O)C2CCN(C(c3ccc(Cl)c(C#N)c3)=O)CCC12 CC1CC=C(C(=O)NCc2ccc(C(=O)N(C)CCc3ccccn3)nc2)CC1 C(C(C)(CCO)NC(=O)CC1CCC(NC(=O)C(n2ccnc2C)C)C1)OC C(CN=c1ccc(C(=O)OC)c(OC)[nH]1)NC(Cc1c(CC)cccc1)=O C(=O)(C(F)(F)C(C)(C)O)NCCOCCN(C)C(C1CC2CCC1O2)=O c1(C(=O)NC2C(CCC)CN(C(=O)C#CC3CC3)C2)nc[nH]c2ncnc1-2 C(=O)(N=c1cc(Cl)nc(O)[nH]1)c1c(CC)nc(-c2ccccc2)[nH]1 c1(C(N2CCC(CCNC(c3cc[nH]c3)=O)C2)=O)nccnc1Cl c1(C(N2CCOCC(NC(c3c(C)nc[nH]3)=O)C2)=O)ccc(C)c2ncccc12 c1(C(=O)N(Cc2cccs2)CC2CCCO2)ccc(C2CCC23CCC3)cc1 C1(C(N2CCC3CCC23)=O)(NC(CSCCC(C)C)=O)CC(C)(C)C1 CCC(C)(CNC(C1CC(C)(F)C1)=O)C(=O)Nc1cncnc1OC O=S1(=O)CC2CN(S(=O)(=O)c3cnc(CO)c(Cl)c3)CC2(NCC2CC2(F)F)C1 c1(C(N2CCC(C(NOC(C)(C)C)=O)C2)=O)ccc(O)nn1 C1(C(C)NC(C2(c3ccccc3F)CCC2)=O)CN(C(=O)OC(C)(C)C)CCO1 c1(C(=O)NC(C2CC(NC(C3CC4(CCCO4)C3)=O)C2)C)cnn2c1CCC2 c1(NC(C2N(C(CC)=O)CC(F)C2)=O)ccc(O)cc1C(F)(F)F N1(CC(=O)N(C(C)(C)C)C)CC(N2CCN(C(=O)O)CC2)C(C)C1 N1(CC(=O)NC2C3(CN(C(C(C)N4CCC4)=O)C3)SCC2)C(=O)CC(C)(C)C1=O CCCCC(C(=O)N1CCC1C(=O)NCC)NC(C1CCC2(CCC2)C1)=O S(=O)(=O)(c1ccc(NCC2=CCCC2)cc1Br)NCc1cc(OC)c(Cl)nc1 C1(OC)CCN(CC(c2cc(C)n(Cc3ccccc3)c2C)=O)CC1C(=O)O C12(CNC(C(C)SCCCC)=O)CC(CN1C(c1ccn(C(C)C)n1)=O)C2 C1(NC(COCCC(C)C)=O)CCC2(CCCN(C(=O)CC(F)(F)C(C)C)C2)C1 C(=O)(C(C)(C)N=[N+]=[N-])N(C)CC1CCCC(C(F)(F)F)C1 C1(C)(C(N(CCCCCNC(C2(CC)CC2)=O)C)=O)CCSCC1 CN1N=CC(CC(N2CC(N(C(=O)Cn3ncc(Br)n3)C)C(O)C2)=O)C1=O C(=O)(C1=Cc2cc(F)ccc2OC1)N(CC(C)NC(C(CC)C(C)O)=O)C Cc1onc(CC(N2CCCOC(CNC(C3(C(F)(F)F)CC3)=O)C2)=O)c1C#N C1(C)(CC(=O)NCCC(C)NC(=O)C(n2cc(Cl)cn2)C)CCOCC1 C1(C(=O)NCCCN(C(=O)CC2(C3CC3)CC2)C)CCN(c2ncccn2)C1 C12(CNC(CN(C)S(N)(=O)=O)=O)CCC(NC(=O)CC3CN4CCC3CC4)(CO1)C2 CC1CN(C(=O)CCC2CCN(C)C2)CC1NC(C1CN(CC(F)(F)F)C1)=O CCC(CC)C(F)C(=O)N(CC(CC)NC(=O)CO)CC c1(NCC(C2CCOCC2)OC)nccc(=NCCC2(CO)CCC2)[nH]1 N1(c2n(CC(OCC)OC)c(CNS(=O)(=O)CC)nn2)CC(CC)C(C)CC1C C1(C)(CNC(Cc2scc(C)c2)=O)CN(C(=O)CCSC2CCCC2)C(C)(C)C1 Cc1nc(C(=O)NCC(C2CC2)N(C)C(c2cc[nH]n2)=O)sc1C c1(C(N2C(C(=O)NCc3ccccc3)CCCC2)=O)ccc2cc(Cl)ccc2n1 CCC(C)CC(=O)NCC1CCN(C(c2cncc(OC(F)F)c2)=O)C1 Cn1ccc(C=CC(N2CC(OCC(=O)NCC(C)(O)CCO)C2)=O)c1 c1(C(N(CCCOCCN(C)C(c2cc(Cl)ns2)=O)C)=O)n[nH]c2cccnc12 c1(OC)ccc(F)c(C(=O)NCCn2cc(C)nn2)c1.C1(O)CCN(C2CCC2)C1 C1(C(N(CCOCCN(C(=O)CNC=O)C)C)=O)CCCC2(CC2)C1 C1(NC(c2c(SC)cc(C)cc2)=O)CC2CCC(C1)N2C(=O)C(C)CCN(C)C N1(C(=O)Cc2cc(F)c(Cl)cc2Br)CC2CC(C2)c2ccc(Br)cc21 N1(C(c2n(CC)ccn2)=O)CCC2CCC12CNC(=O)CCCCC#N Cc1cc(C=CC(=O)NC2(N3CCNC3=O)CC2)ccc1Br c1(C(=O)NCC2(F)CC(NC(c3c(CC)cccn3)=O)C2)cc(Cl)ccc1O Cc1ccc(-n2cc(C)cn2)c(OCCCNC(=O)C(C)CC(N)=O)c1 c1(C(c2nnnn2CCSC)NCC=CC)cccc(C(=O)NCCC)c1 N1(C(C(C(CC)C)OC)=O)CC(O)(C2(CNC(=O)CCC3CC3)CC2)C1 C1(COC(C)C(=O)NC2CC2)CC(O)C(O)CC1C(=O)NCCN(C)C C1(C(=O)OC)CCC(CO)CC1.c12ccc(cc1)OCC(=O)NCCCNC2=O Cc1ccc(CC(N2CCN(C(C3CCCCCC3)=O)C3CC23)=O)cc1[N+](=O)[O-] c1(SC)ccccc1C(=O)NC1(C)CN(C(=O)CN(CC(C)(C)C)C)C1 Cc1nn(C)cc1C(=O)NCC(C)(C)CNC(=O)C(F)CC1CCOC1 N1(C(=O)CN2CCC(F)CC2)CCCC2C1CCN2C(C1CC1C(F)(F)F)=O CN1CCC(OCC(N2CC(O)CC2CNC(c2cccc(CO)n2)=O)=O)CC1 Nc1cc(C(=O)NC2CCC(CNC(C3CCCC34CC4)=O)CC2)ccc1Cl N1(C(CC(C)(C)C2CC2)=O)CC2(CC2)CC1CNC(=O)CN1CCCCS1(=O)=O C1(CC(N2CC(CC(C)NC(=O)Cc3cncn3C3CC3)C2)=O)CCC=CCC1 C1(NC(=O)COc2cncc(Cl)n2)CN(C(C2CC(F)(F)C2)=O)C2(CCCC2)C1 N1(C(C)C)CC(NC(C2(CNC(=O)CCC3CC3(C)C)CCCO2)=O)C(C)C1 c1(C(N2CC(C)C(NC(C3(S(N)(=O)=O)CCC3)=O)C2)=O)ccc2ccccc2n1 N1(C(CCNC(=O)OCC)=O)CC(C)CCC1C(=O)N(C1CCCC1C)C C1(F)(C(N(C(C)CCO)C)=O)CCCN(C(=O)CC#N)C1 c1(C(N2CCC(C)(CNC(CC=C=C)=O)C2)=O)ncc(N)cc1Cl C1(c2cc(CNC(C=NOC)=O)on2)CCN(C(c2ncccc2OC)=O)CC1 CCC(CCC(=O)N1CCC(C)(CCO)CC1)NC(=O)Cc1cscn1 c1(NC(c2csc(I)c2)=O)c(F)ccc(Cl)c1CO c1(C(N2CCC3(NC(c4ccc(Br)s4)=O)C(C2)C3)=O)ccc2c(n1)CCC2 c1(CC(=O)NCC2(F)CC(CNC(C(C)NC=O)=O)C2)ccccc1Cl C(=O)(CC(C(F)F)n1ccnc1)NC1CC(C)(NC(c2c(C)nn[nH]2)=O)C1 c1(N(CCS(CC)(=O)=O)C)ccnc2cc(I)sc12 Cc1cc(C(=O)NCC(CC(C)C)NC(=O)CC2(CO)CCCC2)ncc1C#N CC1Cc2ccc(Br)cc2CN1C(=O)Nc1c[nH]c2cccc(Br)c12 CC1CCN(C(c2ccc(Cl)o2)=O)CC1CNC(c1occc1F)=O C1(CNC(c2cnn(C)c2C(F)(F)F)=O)CC2CCC1N2C(=O)CCCC#N N1(C(C2(NC(C)=O)CCSC2)=O)C2CCC(C2)C1C(N1CCN(C(C)C)CC1)=O c1(C(=O)NC2(CNC(C3=NOC(C)C3)=O)CCCCC2)cc(C#N)c(F)cc1F N1(C(CC(CC)OC)=O)CC(C(=O)NCc2cc(C)cnc2O)CCC1C C#CCC(C)(C)C(=O)NCC(=O)NCC1CC(C)N(C(c2cc(C)nn2C)=O)C1 N1(CC(=O)NC2(CF)CCN(C(C(CCC)OCC)=O)C2)C(=O)CC(C)(C)C1=O C1(CCNC(C2(F)CC(C(=O)OCC)C2)=O)(OC)CN(C(C2(C)CCCO2)=O)C1 C12(C(=O)NCC(C)(C)OCCNC(c3csc(Cl)c3)=O)COCC1C2 c1(CCC(=O)NCCSCC)cn(C(C)C(N2CCOCC2)=O)nn1 c1(NC(CSC)Cc2cccs2)cc(=O)n(CC(=O)O)nc1Cl CC(=O)CCCC(=O)N1CCC(C(=O)NC2CC(CF)C2)(C(C)C)C1 C(=O)(C(CCO)N(C)C)N(CCCNC(C(C)(C)N(C)C)=O)Cc1ccccc1 C(=O)(CC(C)CC(C)C)N1CCC(O)(C(C)NC(C(Br)=C(C)C)=O)CC1 C(=O)(CC(C)P(C)(C)=O)N1CCC(C(CNC(C2=C(C)CCC2)=O)(C)O)CC1 C=CCC(F)(F)C(=O)NCCCC(C)NC(=O)Cc1csc(C(C)C)n1 c1(NC(c2cc(Cl)sc2Cl)=O)cnc(F)cc1C(=O)NCCN(CCO)CCO C1(NC(=O)CC2CC3(CC3)C2)CCN(C(=O)C(F)n2cccn2)CC1F c1(C(=O)NCC2CN(C(c3cc(C)c(C)[nH]3)=O)C(C)C2)c(C)nc(C)n1O C(c1ccc(F)cc1)=CC(N1CCC(CCNC(C(COC)OC)=O)C1)=O N(C1CN(C(=O)CCC(F)(F)F)Cc2ccccc21)C(C(C)c1cccs1)=O Cc1cc(C(=O)NCC2(CCNC(=O)C(C)NC(=O)CC3C=CCC3)CC2)c[nH]1 N1(C(C(C)(C)C)=O)CCCCC1C(N1CCC(CNC(c2cnc(O)s2)=O)C1)=O N1(C(c2c(CC)cco2)=O)CC2CCN(C(=O)CCC(=O)OC)CC12 c1(CN(CCN(C)C)C(=O)NC2(Br)CC2(F)F)cccnc1 c1(C(N2CCCN(C(C(CCC)(C)C)=O)CCC2)=O)ccc2nc(=N)[nH]n2c1 C1(C(CC)C)CCN(C(c2cccc(CN(C)C(c3cccs3)C)c2)=O)CC1 C1(CC(=O)Nc2ccccc2Cl)C2CCC(C2)N1C(=O)Cc1cccc(F)n1 C1(CNC(C2(C#N)CC2)=O)CC2(CCN(C(=O)COc3ccccn3)CC2)CO1 c1(C(C)C)cc(C(=O)NC23CC(NC(=O)CC#N)(C2)C3)n[nH]1 c1(OC(C(N2CC(=CCNC(CSCCC(C)C)=O)C2)=O)F)ccc(Cl)c(F)c1 C=C=C(C)CC(=O)N1CC2CC2(NC(c2sc(Cl)cc2Cl)=O)C1 c1(N2CCC(N(C(C(C=C)O)=O)C)C2)nc(C)cc(C(F)(F)F)c1C#N c1(CNC(C2CCC(C)N(C(=O)Cc3cncn3C)C2)=O)cnc2cc[nH]c2c1 CCCCCCCCNC(=O)C(=O)NC1CC1C(=O)NC(=O)CCc1ccon1 C1(C(=O)NC2CC2)CSCN1C(=O)C(c1ccccc1)F Cc1c(F)ccc(C(=O)NC2CCN(C(c3ncccc3Cl)=O)C2C)c1C C=CC1(NC(c2ccn3ccsc23)=O)CCN(C(=O)OC(C)(C)C)C1 c1(C(N(C(CNC(C=CC=CC)=O)C)C)=O)cn(C(C)C)cc1C c1(CC(N2CCC(N(C(C3CCCCS3)=O)CC)CC2)=O)noc(C)c1C#N C(=O)(C(F)C(F)(F)F)NCC(CC)(C)NC(=O)CNC(C1CCC1)=O c1(CCC)c(C(=O)NC23CC(C2)N(C(=O)Cc2sccc2C)C3)cnn1CCO C1(NC(C(c2cccc(C)c2)C)=O)CCN(C(c2n[nH]c3c2COC3)=O)C12CC2 c1(C(=O)NCCCC#C)ccc(CNC(c2ccc(OC)nn2)=O)nc1 C12(C(=O)NCC(C)NC(C3(C4CCCCO4)CC3)=O)CCCN(CC1)C2 C1(CC(=O)N(CCCOC)CC(C)C)CC(NC(c2cn[nH]c2)=O)C1 N1(C(C(C(C)C)(C)C)=O)CC2CC(NC(=O)CC(C)(O)C3CC3)CC2C1 C1(C(=O)NCCCN(C(c2ccc(C3CC3)cn2)=O)CC)CCS(=O)(=O)N1 N1(C(C2CC(CC)N(C(c3csc(C#N)c3)=O)CC2)=O)CCS(=O)C(C)C1 CC(C)C(CC(=O)N1CC(NC(=O)C(=O)N(C)C)C1)C(C)C Cc1nn(C)c(C)c1CC(C)C(=O)NCC(C)NC(=O)CNc1ccc(Cl)cc1 CC1CC(=O)NCC1C(=O)N(C1(C(=O)NCCC2CC(F)(F)C2)CCC1)C1CC1 C12(NC(c3csc(Cl)c3)=O)CCN(C(=O)CCCCc3ccccc3)CCC1C2 N(C1CCCc2n[nH]cc21)C(C(CC(C)(C)NC(CC(C)c1ccco1)=O)F)=O c1(CC)cc(C(N2CCOCC2C2CCOC2)C(=O)NC2CCOC2)cc(C)c1 C1(NC(c2sc(F)cc2Cl)=O)COCCN(C(=O)CCN2CCCCCC2)C1 c1(C(N2CC(C)C(NC(=O)CC3CC3)C2)=O)nn(C)c(=O)c2ccccc12 C1(NC(c2c(C(C)C)noc2)=O)CC2CCC(C1)N2C(=O)C(C)n1cnnn1 N1(C(c2cnn(C(C)C)c2N)=O)CC(C)CN(C(=O)CCc2cnc[nH]2)CC1C C(=O)(C1=NOC(COCC)C1)N1CC(N(CCC)CC)C1.c1(C(=O)N)nccs1 c1(CC(=O)NCC2(F)CCN(C(COC)=O)C2)cccc2c(C)csc12 c1(C(=O)NC2(CO)CCN(C(c3[nH]c(CC)c(Cl)n3)=O)C2)nccc2[nH]ccc12 N1(C(CC2(C)CCN(C(C(CC=C)NC(C)=O)=O)C2)=O)CC2CC3CC2C1C3 C1(C(N2CCN(C(C3(C#N)CC(C)C3)=O)CC2)=O)(CC)CCNC1=O c1(NC(=O)NCC(N2CC(NC(=O)C(Cl)=CCl)C3CC23)=O)ccccc1C1CC1 C=C1CCC(C(=O)NCC2CC2CNC(=O)C(c2ccccc2)N(C)CC)CC1 C1(Cn2cc(C3(C)CCOC3)nn2)CCN(C(c2nc(Cl)cs2)=O)CC1 c1(C(N2C(C)(C(=O)Nc3cccc(F)c3CO)CCC2)=O)cc(F)c(F)cc1O C1(COC)(CNC(=O)Cc2cnoc2)CN(C(C2(NC(N)=O)CC2)=O)C1 c1(OC)cccc(CNC(=O)CNC(=S)Nc2cccc(F)c2)c1 c1(COC)ccccc1C(=O)NC1CCCCC1CNC(c1nc(O)c(C)s1)=O N1(C(c2n(C)cnc2)=O)CC(C)(CNC(c2cnc(C3CCC3)o2)=O)CC1(C)C Cc1cc(C(=O)NC(C2CCN(C(=O)CSc3nccn3C)CC2)C)nc(O)n1 C1(NC(Cn2ncc(C)c2)=O)C(C)CN(C(c2cc3cnccc3o2)=O)CC1C Cn1ccc(CC(=O)N(C(=O)CCC2CCC(=O)C2)CCCN(C2CC(=O)C2)C)c1 C(=O)(C1c2c[nH]nc2CN1C(c1ccn(C2CC2)n1)=O)NCC(COCC)C CC1(CNC(=O)CSc2nnnn2C)CC(NC(C2(CS(C)(=O)=O)COC2)=O)C1 c1(C(=O)NCC2CC(NC(C(CC)CC)=O)C2(C)C)cc(F)c2ncccc2c1 C(=O)(C(C)(C)C(=O)NCCC1CC(NC(=O)Cc2nc[nH]n2)C1)OC C(=O)(CC1=NNC(=O)C1)NCC(N1CCN(C(C2(COC)CC2)=O)CC1)=O c1(CC(=O)NCC(C)CN(C)C(C2CC(C)OC2C)=O)cccnc1Cl n1(CC=C)cc(-c2cscc2CN(CC(C)C)C)cn1 C1(c2nc(CNC(C3(CC)CCCC3)=O)[nH]n2)CCN(C(C2CC2(Cl)Cl)=O)CC1 N1(C(=O)NC(C2CCCC(C)C2)(C)C)CCNC(=O)CC1 c1(C(=O)NC2C(CNC(C(CSC)O)=O)CCC2)cc2ccccc2cn1 CCCC(C(=O)OC)C(=O)NCC1CC(C)CCN1C(c1csc(C)c1)=O C1(N(C(=O)Cc2ccccc2Cl)CCC)CCN(C(=O)Cc2ccsc2C)CC1 Cc1ccc(N)c(C(=O)NC2C=CC(CNC(c3cc4n(n3)CCO4)=O)C2)c1F C1(NC(CCc2n(C)c(S)nn2)=O)CN(C(=O)Cn2cccc2)C2(CCC2)C1 c1(C(=O)NC(C(C)NC(C(CC)n2nccc2C)=O)CO)cc(SC)nn1C CC1CN(Cc2cocn2)CCN1C(c1cc(I)ccc1F)=O N1(CC(N2CCC(N(CC#C)C(c3cnc(Cl)s3)=O)C2)=O)C(=O)CC(C)(C)C1=O O=C1CCC2CN(C(C3CC(=O)C3C(F)(F)F)=O)CC2N1 c1(OC)ccnc(C(N2CCCC(N(CCO)CCN(C)C)C2)=O)c1OC S(=O)(=O)(c1ccc(NC2CCCC2)cc1Br)NC1CCC(NC(N)=O)C1 CP(C)(=O)CN1CC(C(=O)NC2CC(NC(C3C4CC5C(C4)C35)=O)C(O)C2)C1 c1(CCC(=O)NC(c2cn3ccccc3n2)C)ccc(C#N)cc1F CC(C)CCCCC(=O)NCCCOCCN(C(=O)CCC1(C)CCC(=O)N1)C c1(NCC(n2ccnn2)C)ncccc1S(=O)(=O)NC(CC1CCCC1)CO C1(N(C(c2ccc(C#C)cc2)=O)CC)CC12CCN(C(=O)Cc1nc[nH]n1)CC2 c1(C(=O)NC23CC(CNC(c4ncc(F)cn4)=O)(C2)C3)cnc2nccn2c1 c1(OCC(=O)NC(C)CCNC(=O)C(C2(O)CCCC2)F)cccnc1 CN1CCN(C(C2CCC(O)CN2C)=O)CC1CNC(c1ccc(F)cn1)=O CCC(CC(=O)N1CC(O)(CCNC(=O)CC(=O)OC)C1)C(C)C Cc1cc(C(=O)NCC(C)N(C)C(c2cc[nH]c2)=O)cc(Br)c1C C(=O)(C1=CCS(=O)(=O)C1)N(C1CN(C(CC2CN(C)CC2O)=O)CC12CC2)C C1(NC(=O)C=Cc2cnc[nH]2)COC2(C1)CN(C(=O)COc1ccc(Cl)cc1)C2 c1(C(=O)NC2C(C)N(C(c3cc(F)ccc3Cl)=O)CCC2)ccc2nccn2c1 c1(C(=O)NC2CC(N(C(C3C(CC)C3)=O)C)C2)cc(-c2cccs2)on1 c1(CC(N2C(C(=O)NC(COC)CO)CC2)=O)csnc1C c1(CC)nn(C)cc1C(=O)NCCOCCC(=O)NCC(C(C)C)OC C12(NC(C(C3CCC3)OC)=O)CC(NC(c3n[nH]cc3C)=O)(C1)C2 N1(C(=O)OCC)CCC(C)CC(NC(=O)Nc2ccc(CSC(C)(C)C)cc2)C1 Cc1ncc(C(=O)NC(CCNC(C2CCCC23CCC3)=O)C(C)C)cc1C#N O=C(N=c1[nH]nc(O)s1)C1=NOC2(CCN(C(c3cc4c(s3)CCC4)=O)CC2)C1 C(=O)(C(C)(C)C(F)(F)F)NCC(CC(C)C)NC(C1CCn2nnnc2C1)=O CC1CCSCCN1C(C1CCN(C(c2cc(O)cc(=O)o2)=O)CC1O)=O N1(C(C2CN(C(C)=O)C2)=O)CCN(C(=O)CC2CN(C)CC2O)CC1C(F)F c1(C(N(CC(F)(F)F)CC=C)=O)cn(C(F)F)nc1C(F)F C1(NC(COCCC)=O)CCN(C(=O)C(C)Cn2cccn2)C12CC2 Cc1ccc2cc(C(=O)N(CC(C)NC(=O)CN3CCCC3C)CCO)[nH]c2c1 N1(C(CN(C)CC)=O)CCN(C(c2cc(Cl)no2)=O)CC1c1ccccc1OC Cc1cc(O)ncc1C(N1CCC(C(=O)NC2COC3(CCC3)C2)(CO)C1)=O c1(CCC(=O)NCCC2CC(NC(C3C(C=C)CC3)=O)C2)ccc(SCC)cc1 CCCC(CCC)C(=O)NC1CC2CCC1N2C(=O)CC(C)(C)COC(C)=O c1(OC)nn(C)cc1C(=O)NC1CCC1NC(c1cncc(N)c1)=O C1(NC(c2cc(=O)cc(Cl)[nH]2)=O)CCN(C(=O)Cc2ccsn2)CC(O)C1 C=C(C)CC(C)C(=O)N1CC(N2CCN(C(C3CC(C)(O)C3)=O)CC2)C1 C1(CNC(CC=C(C)C)=O)OCCC1C(=O)N(CCCc1ccco1)C C#CCCCCC(=O)N1CCC(F)(C(=O)NC(c2cccs2)C)CC1 N1(C(c2c(C)nc(C3CCC3)o2)=O)CCCC2CN(C(=O)C(C)CN(C)C)CC12 c1(CCCCNC(C(CC#C)C2CC2)=O)cc(O)ccc1C C1(C(=O)NC(c2ccncc2)CC)CCN(C(c2cccn2C2CC2)=O)C1 C1(C)(CNC(CCCC(C)O)=O)CC(F)(F)CN1C(c1ncc(Cl)n1C)=O c1(C(=O)NCCCN(C(c2cc(N(C)C)ccn2)=O)CC)nc(O)c(C)s1 c1(NC(C2C(CNC(C(CCC)C#N)=O)OCC2)=O)ccn2nccc2c1 CCC(CC)CC(F)C(=O)NCC1CC1C(=O)Nc1ccc(C)cc1F c1(NCC2(COC)CCNCC2)cnc2n1CCCC2 C(c1ccc(F)nc1)=CC(N1C(C)CC(NC(=O)CCc2ccc(Cl)nc2)C1)=O N1(C(COC2(C)CCCC2)=O)Cc2ccccc2C1CNC(C1CCC1(F)F)=O Cc1cnc(NC(c2ccccc2)=O)nc1.c12cccc(c1)NCC2=O c1(C(C)NC(C(C2CC=CCC2)NC(CC(C)C)=O)=O)cccnc1O C1(CC(=O)NCC(C)(C)OCCNC(C2(F)CC2)=O)CCNC1=O c1(-c2cn(CC(C)NC(CCNC(=O)OC)=O)nn2)ccnc(OC)c1 C12(C(=O)N(C(C)C3CC3)C)C(NC(C3CCC3C#N)=O)C3CC1C2C3 N1(Cc2ccc(OCC)cc2)CCC2(CC1)CC2C(N1CCC2CCCC2C1)=O C(=O)(C(C(C)O)NC(C1CCCC1CNC(C1CCCC(=O)C1)=O)=O)OC O(S(=O)(=O)c1c(C)nn2cccnc12)c1cc(C)c(Br)cc1 n1(CC)ccc(CC(=O)NC2CC2CNC(=O)C(COC)Sc2ccccc2)n1 c1(OC)ccc(C(N2CCCC(C)(CO)C2)C(=O)NCCCSC)c(C)n1 C1(NC(c2cc(C(F)F)[nH]n2)=O)CC12CCN(C(=O)Cc1ccc(Cl)cc1)CC2 C1(N(C(=O)CCCc2ccccc2)C)CC(CNC(C)(C)CC2CCC2)C(O)C1 N1(C(C2(SC)CC2)=O)CCc2ccccc2C(NC(c2ccn(C)c2C)=O)C1 c1(C(N2C(CNC(C=C(C)C)=O)CCC2)=O)cc([N+](=O)[O-])ccc1Cl N1(C(C(C2CCCC2)OCC)=O)CCC2(CCCN2C(c2ccc(C#N)o2)=O)C1 N1(C(C(C)OCC#C)=O)CCCC(C)(C)C1C(=O)NC1(c2ncccn2)CC1 c1(CN2C(CNC(C3C(C)OCCC3)=O)CCC2)ccc2c(c1)CCC2 c1(C(=O)NC2C(C)(C)CN(C(=O)C(O)P(C)(C)=O)CC2)cccc2cnccc12 c12cncc(c1)NC2=O.N1(CCOCCC)CCC(Cn2ccnn2)C1 C1(NC(C(N2CCNC2=O)C)=O)CCOC12CCN(C(c1ccc(Cl)s1)=O)CC2 C(=O)(CS(=O)(=O)c1ccccc1C)NC(CC)(C)CNC(C1(CN(C)C)CC1)=O C1(NC(CCCc2ccc(C)cc2)=O)CN(C(C2CC2CF)=O)CC2(CCC2)C1 CC1N(C(c2conc2CNC(=O)C=C2CCOCC2)=O)CCOC1(C)C C1(C(=O)NCCCC)CCC(CNC(=O)COC2CCCC2)C1 N1(C(c2ccc(C)cc2Cl)=O)C2CCC1CN(C(=O)Cc1occc1C)C2 C1(C=C)(CC(=O)NCc2scc(CNC(C(C=C)(C)C)=O)n2)CCOCC1 c1(CC(=O)NCC2(OCC)CN(C(CS(CC)=O)=O)C2)ccc(Cl)c(C)c1 c1(OC)ccc(CC(=O)NCC2CCCCN2C(c2cccnn2)=O)c(OC)c1 c1(C(=O)NCC2(CCNC(C(C)OCC#C)=O)CC2)c(F)ccc(OC)c1N C1(CNC(CNC(CC)=O)=O)CC2CN(C(C3CNC(=O)N3C)=O)CC12 N1(C(CCN(C)CC)=O)CCCN(C(c2cc(N3CCCC3)ccn2)=O)CC1C c1(C(=O)NCC(C)(C)CNC(=O)C2=CCCOC2)c(C(F)F)nc2ccccn12 CCC(C)(C)C(=O)C(=O)N1CC(F)(F)CC1(C)CNC(=O)Cn1cccn1 C1(NC(CCC2C(C)C2)=O)C2CC1CN(C(C1(O)CCOCC1)=O)C2 C(N=c1[nH]c(Cl)nc2[nH]ccc12)NC1CCN(C(=O)CS(=O)(=O)C2CC2)C1 C1(CC(=O)NC(C)(C)CC2CCOC2)CN(C(=O)CC2CC3(CC3)C2)CCO1 CC(C)(CF)C(=O)N1CCC(N2CCN(C(c3cnc(=N)[nH]c3)=O)CC2)C1 c1(C(N(C)CC2N(C(CC(C)F)=O)CCC2)=O)cnnc(O)c1 CS(=O)(=O)CCNCC(N1CCCC1CO)=O N1(C(C(=O)NCCOC)=O)CC2CC2(NC(=O)Cc2csc(CCC(F)(F)F)n2)C1 C1(C2CCOCC2)(NC(C2N(C(C(C(=O)OC)C)=O)C(C)C2)=O)CC1 C1(NC(=O)C2CC2)CC2(CCN(C(C3C(C4CC4)C3(F)F)=O)CC2)C1 Cc1cc(N2CCN(CCCNC(c3csc(C4CC4)n3)=O)CC2)nc(CO)n1 c1(CC#N)ccc(OCC(N2CC(N3CCN(C(=O)CC#N)CC3)C2)=O)cc1 c1(OCC)ccc(CCC(=O)NCC(C2CC2)NC(C2(C3CCC3)CC2)=O)cc1 Cc1nc(-c2ccccc2)oc1C(=O)N(C1CCN(C(C2CC2C2CC2)=O)C1)C c1(C(=O)OCC)csc(-c2nc[nH]n2)n1.C1(CN2C(=O)CC3C(C3)C2)CCCO1 c1(C(=O)NC2C(NC(C3CC(C)(C)C3)=O)COCC2)cc2cnccc2o1 C=CCC(C)(C)C(=O)N1CC(C(C)(C)O)(CNC(C2CCC(=O)N2C2CC2)=O)C1 C12(NC(=O)COCc3nc[nH]n3)CCCC1CN(C(=O)CCc1ccncc1)C2 C(=O)(C1CCc2cc(F)ccc21)NCCCN(C(c1cnc(CCCC)s1)=O)C C#Cc1cncc(C(N2CC(C)CC(O)C2)C(=O)NC2CCOC2)c1 CC1(C)CC2CC(C)(CN2C(C(=O)NCCC2CC2)c2cnc[nH]2)C1 c1(C(=O)NC2CC(C)(CC)C2)cncc(C(=O)NC(C2CN(C(=O)NC)C2)=O)c1 N1(C(CSCCOC)=O)CC(NC(c2nccn3nccc23)=O)CC2(CCC2)C1 Cc1cc(C)n(CC(N2CC(NC(c3cc(-c4ccco4)c[nH]3)=O)C(O)C2)=O)n1 Cc1oc(CO)cc1C(=O)NCc1cnn(C)c1C(=O)NCCC1CC1C C(CCCCNC(=O)C(N)=O)N(c1ccccc1)C(CN(CC)CC)=O c1(C(=O)NC(CN(C(C(C)(CO)OC)=O)C)C)cc2c(nc1O)CC(C)(C)CC2 C(C(C)C(=O)NC(C)(CNC(c1ccc(CNS(C)(=O)=O)o1)=O)CC)OCC N1(c2ncc(OC)cn2)CCC(F)(F)C(C(=O)NS(=O)(=O)CCSC)C1 C(=O)(C(F)(F)c1csc(Cl)n1)NC(C)C(C1CCCCC1)NC(=O)C=CC1CC1 c1(NC(C(c2nccs2)N(C)CCNC(C)(C)C)=O)ccc2c(c1)OCO2 c1(C(C(=O)NCCCC)N(CC(F)(F)F)CC2CC2C)ccc(CC(=O)OC)s1 CC(C)(CS(C)(=O)=O)C(=O)NCC1CCC1NC(c1ccnc2ncnn12)=O C1(NC(C(C)c2ccco2)=O)CC2(CCN(C(=O)CC(C)(C)F)CC2)C1 CCCC(CC)C(=O)NC(Cn1cncn1)C(=O)NCCCN1CCCC1=O C1(C(=O)Nc2c(CC)nn(C)c2)CCN(C(=O)CC2=CCN(C)CC2)O1 C1(NC(CC2(OC)CCCC2)=O)CCC2(CC1)CN(C(C1CC1F)=O)CCO2 CCCCCCCCCCC(=O)NC1(C)CCN(C(C2CC(C)CO2)=O)CC1 N#Cc1cnc(NC(C2(O)CCN(C(c3c(Cl)cccc3I)=O)C2)=O)c(Cl)c1 N1(C(CCOCCOC)=O)CCC2(CCN(C(=O)C(CC)C(=O)OC)C2)C1 c1(C(=O)NC2CC3N(C(CC(=O)OC)=O)C(CC3)C2)ccc(Br)c([N+](=O)[O-])c1 c1(C2CC(CC(=O)OCC)(NS(=O)(=O)CC3CCC(C#N)C3)C2)cccc(Br)c1 c1(OC)cc(C)c(S(=O)(=O)NC(=O)C2=CCCN(S(=O)(=O)C(C)C)C2)c(C)c1 C12(C)CC13CCN(CC3)C2=O.c1(NC(=O)OC(C)(C)C)ccc(C#N)cn1 C1(NC(C(C(=O)OC)OC)=O)CCCC12CN(C(c1cc3cccnc3s1)=O)C2 N1(C(CCN(CCOCCOC)C)=O)CCN(C)C(CNC(=O)CC)C1 c1(C(=O)NCC2CCCN(C(C(CCSC)O)=O)CC2)n[nH]c2c1CCSC2 C1(OC)CCC(c2nnnn2C2CC2)(NCC2(c3cc(F)ccc3F)CC2)CC1 C1(CNC(CC2C(C)=NOC2=O)=O)CN(C(=O)CC(=O)NC2CC2)CCC1(C)C c1(CN(C(c2c(C)nc[nH]2)C(=O)NC2CCOCC2)C)cccc(C(C)(C)C)c1 N1(C(Cc2cc(CC)no2)=O)CCN(C(=O)C(C)OC2CCCCC2)CC1C1CC1 C1(CNC(C(CN(C)C)(C)C)=O)CCC(C)(C)CN1C(C1CC(F)C1)=O CC(C)C1C(=O)N1.c1(C(=O)OCCCCCc2ccccc2)ccc(N)cc1 C1(NC(C(CCC)OCC)=O)CCC2CC1CN2C(c1nncn1C)=O c1(C(=O)NC23CCN(C(Cn4c(C)c(Cl)cn4)=O)CC2C3)ccc2c(c1)COC2 c1(C(=O)OC)ccn2c1CN(C(C(=O)N(C(C)(C)C)C1CC1)c1cnsc1)CC2.C(=O)O N1(C(C2CCCC23CCC3)=O)CC2CN(CC3CCOC3)CC2C1 N1(C(CN(CC(C)(C)C)C)=O)CC=CC(NC(=O)C(O)C(F)F)C1 Cc1ccc(F)c(N)c1C(=O)NCC1C2CCC(C2)N1C(=O)Cc1ccns1 N1(C(c2c(CC(=O)OC)occ2)=O)CCN(C(c2cccnc2)=O)CC12CC2 CN(Cc1ccc(S(=O)(=O)N(C)C)cc1)N1CC(S(C)(=O)=O)CCC1C c1(C(=O)NC(CC2CN(C(C(=O)NC(C)C)=O)C2)C)cnc(CC2CC2)nc1 C1(NC(Cc2scc(C)n2)=O)CCCC12CN(C(=O)Cc1cncn1C)C2 CON1CC(C(=O)N(CC(=O)NCC(C)(O)C(F)F)C2CCC2)CC1=O c1(CC(=O)NCC2(NC(C3(C(F)(F)F)CC3)=O)CCCC2)ccc(F)c(SC)c1 N1(C(C(C)(O)C2CC2)=O)CCC2CC(NC(c3cccc[n+]3[O-])=O)CCC2C1 CC1(C)OCCOC1C(=O)NC1CC(F)CN(C(C2CCSCC2)=O)C1 c1(OC)cc(CC(=O)N(CCC(C)NC(=O)C(C)NC(=O)C(C)(C)C)C)ccn1 c1(C(=O)NC2CCN(C(C(CC3CCC3)NC(C)=O)=O)C2)cnc(=N)[nH]c1 C1(CNC(C2CCC2)=O)CN(C(=O)CC2CC3(CC3)C2)CC(C(F)(F)F)O1 c1(OC)ccc(C(O)C(C)N(C(=O)C=CC=C(C)C)C2CC2)cc1 C1(=O)C(C(C)C)C(=O)N1C1(C(C)O)CC1.c1(C2CCCO2)ccncc1 CS(=O)(=O)CCC(=O)NC1CCCC(NC(c2cc(-c3ccco3)cs2)=O)C1 N1(C(C(CC)=CCCC)=O)CC(N(C(=O)CC=C(Cl)Cl)C)C(C)(C)C1 c1(-c2cc(COC)[nH]n2)nc(-c2cccc(Br)n2)nn1CCN(C)C N1(C(C2CC=C(C)CC2)=O)CCN(C(C2OCCN(C)C2=O)=O)CC(C)C1 c1(C(=O)NCC2(O)CCCN(Cc3cccc(C)c3F)C2)csc2ccccc12 CC(C)CC(CN=c1nc(C2CCOCC2)[nH]s1)NC(=O)C1=CC2CCCC12 c1(C(=O)NC2CCC(CNC(CSCCCC)=O)C2)cc2c(C)n[nH]c2cn1 C(CC(N)=O)(C(=O)NC1CNC(=O)OC1)NC(c1n(CC)ccc1)=O CCCC(C)(O)C(=O)NC1C2CN(C(C3(n4cc(Br)cn4)CC3)=O)CC12 C1(NC(C(CC)(C)CC)=O)CN(C(C2CCCN2C)=O)C2(CCCCCC2)C1 Cc1onc(C2CC2)c1C(N1CC2CC1C2CNC(=O)C(C)n1cnnn1)=O N1(C(C(C(=O)OC)OC)=O)CCn2nc(CNC(c3ccccc3)=O)cc2C1 C1(OCC)CN(C(=O)C(=O)NCC)CC1NC(=O)C(C)OCC(F)(F)F CC(C)CC(CC(=O)NC1(c2cc[nH]n2)CC1)NC(=O)C(C)(O)C1CCC1 Cc1cc(Cl)ccc1C(=O)NCC1(O)CN(C(=O)CC2CCCC2(F)F)C1 C(=O)(CCCCc1cccc(O)c1)N(CC(C)NC(C1CCCO1)=O)C CCC(C)(C)C(C)CC(=O)N1CCC(CCCC(=O)CP(C)(C)=O)CC1 Cc1ccc(C=CC(=O)NCC2CN(C(=O)CCC(F)F)CC2(C)C)c(C)c1 C1(C2CCN(C)CC2)(C(N(CC(CN(C(=O)Cc2ccon2)C)O)C)=O)CC1 N#Cc1ccc2oc(C(N3CCC4(CC3)CC(N3CC(CC#N)C3)C4)=O)cc2c1 C(=O)(CS(=O)CCC(F)(F)F)N(CC(CNC(c1nccc(CC)c1)=O)O)C c1(C(=O)NC2CCN(c3snc(CC)n3)C2)ccc2c(c1)C(C)C(C)O2 C1(C(N2CC(C(C)OC)C2)=O)CC2CC1CN(C(C1CC(O)C(F)C1)=O)C2 C=C(C)c1cc(C#N)ccc1NC(=O)NCc1cc(C)cc(F)c1 Cc1cc(F)cnc1C(=O)NCC1CCCCN1C(=O)CCC(=O)N1CCCC1 C1(F)(CNC(CCN(CC)CC)=O)CCN(C(C23CC(C2)C3)=O)C1 N1(C(C2(OC)CC2)=O)CCN(C(c2cncc(C(F)F)c2)=O)C(C(C)C)C1 N1(C(CN(C(C)C)C)=O)CC2CC(CNC(C3CC(=C4CCC4)C3)=O)C(C2)C1 Cc1cccc2c1CCN2C(=O)C(N1CCCCC(N)C1)=O N1(C(CCOCCOC)=O)CCCCC(NC(c2ncc(Cl)cc2Cl)=O)C1 C(CCN=c1[nH]c(=NC2CC3CC4C(C3)C24)[nH]c2c1CC(C)CC2)OC c1(NC(CC2CN(C(=O)Nc3ccc(OCC)cc3)C2)=O)cc(Br)c(F)cc1F C=CCC(C(=O)N1CCC(C)(CNC(c2cc(Br)n(C)n2)=O)C1)NC(C)=O Cc1cnnc(O)c1C(=O)NCc1c[nH]nc1C(N1CCSC(C)C1)=O N1(C(C2N(C)CC(F)C2)=O)CCCC(O)(CNC(c2ccoc2C2CC2)=O)CC1 C1(NC(=O)CCc2ccc(O)nc2)CCN(C(=O)Cc2cnccn2)CC1CO C(CN=c1[nH]ccc(=NCC2(C)CCCC2O)[nH]1)c1nnc(C)s1 C(CC(O)C(=O)NCC1(c2ccon2)CC1)NC(=O)CC1CCCOC1 C(=O)(C(O)CN(C)C)NCC(=C1CN(C(CC2CN(C)C2)=O)C1)F CCCCCC(CC)C(=O)NC(C)CCNC(c1nn(C)cc1C(F)(F)F)=O C1(C(=O)NC(CC(C)C)CNC(c2c[nH]nc2Cl)=O)CCCCC12CC2 C1(C(=O)NCc2ccc(SC)o2)CCCCN1C(C1(O)CCSCC1)=O C1(C(N2CCC(C)(F)CC2)=O)CC2CCCC2N1C(C1CC1C(F)F)=O N1(C(c2ncc(OCC)nc2)=O)CCCC(NC(C2CCCC2OC)=O)C1C Fc1c(C(F)(F)F)ccnc1CCNCCc1ccsc1 c1(C(N(C)CC2CCN(C(C3(CF)CC3)=O)CC2)=O)cc2ccccc2cn1 N1(C(CCCN(C(=O)OC)C)=O)CCC(CNC(c2ncsc2C)=O)C12CC2 N1(C(Cn2c(C(C)C)nnn2)=O)CCCCC1CN(C)Cc1cccc(O)n1 C1(NC(c2n(C)nc(C(F)F)c2)=O)CCN(C(C2CN3CCC2CC3)=O)CC1O C1(NC(c2ccc[nH]2)=O)COCCC1NC(C1(C(=O)NC2C(CF)C2)CCC1)=O C1(NC(C=CC(CC)C)=O)CCC2(CC1)CN(C(=O)Cc1csnn1)CCO2 Cc1cc2c(cc1C)OC(C(N1CCC(CNC(=O)C(F)(F)CO)CC1)=O)C2 C1(NC(C2CCC23CCC3)=O)CCCCN(C(=O)CSc2ccc(Br)cc2)C1 C(CCCOC)(C(=O)NCCCSC)N(C1CCN(C)C1)CC N1(C(C(c2cccc(Cl)c2)N(C)C)=O)CC(NC(c2ccc(Cl)cc2)=O)C(O)C1 C1(NC(=O)OC(C)(C)C)CC2(C1)CC(C(=O)NC1CCC1)C2 c1(CC(=O)NCC2CC(NC(CC3(C)CC3F)=O)C2)n[nH]cc1Br C1(C)(CN(C(=O)CCN(C(=O)CCCC2CCCC2)CCO)C)C(C)(C)C1(C)C C(C)(C1OCCc2sccc21)NC(=O)NC(c1ccccc1N(C)C)C c1(C(=O)NCC(C)NC(C2(C)CC2(F)F)=O)ccccc1C#N c1(N2CC(C(=O)NCc3ccc(F)cc3Br)C(O)CC2)ncc2cc(Br)cnc2n1 c1(C(N(CC(C)NC(=O)CC2CC2(C)C)C)=O)ccncc1F Cc1ccc2ncc(C(=O)NCC(C)NC(c3cc(CO)n(C)n3)=O)n2c1 C1(C(N2CCC(O)(CCNC(C3(F)CC3)=O)C2)=O)CCc2nn[nH]c2C1 Cc1nc(F)ccc1N(C1CCNCCC1C)C(c1cc(F)c[nH]1)=O C(=O)(C(O)C(C(C)C)OC)N(CCCNC(c1ccsc1C(F)F)=O)CC N1(C(CNC(C(CC)COC)=O)=O)CCOC2COCC12 c1(C(N2C3CC(NC(CNC=O)=O)C2CC3)=O)ccc2c(c1)OCCO2 c1(C(N(CCCN(C)C(C2CCCC2(C)C)=O)C)=O)ccc2cncn2c1 CC1CN(C)CC1NC(=O)C(C1CC=CCC1)NC(c1ccnnc1O)=O c1(N2C(CNC(C(CCC)CCC)=O)CC3(CC3)C2)cc(C#N)ccc1[N+](=O)[O-] C1(NC(CCCCNC(C23CCC(OC)C2C3)=O)=O)CC(C)N(C)CC1C c1(OC)nc(C)ncc1C(=O)NC1(CO)CCCN(C(C2(S(C)(=O)=O)CC2)=O)C1 S(=O)(=O)(c1ccc(NCc2cc(OC(C)CN(C)C)no2)cc1Br)OC(C)(C)C N1(C(CC)C(=O)NC(C)Cc2ccc(Cl)cc2F)CCc2ccccc2C1 CCC(C)C(O)CNC(=O)CSc1ccccc1OCC Cc1nc(SCC(=O)NCC(C)CNC(C2(O)CCC2)=O)n[nH]1 C(c1ccccc1)=C(C)C(N1CCC(C(C)(C)NC(=O)COCC2CCC2)C1)=O Cc1nnc2n1C(C(=O)NCC1CN(C(=O)C3CCCc4nc[nH]c43)C1)CC2 C1(NC(C=CSC)=O)CC2CC(C1)N(C(=O)Cc1noc(C)c1C#N)C2 C1(OCCNC(C)C(C2CCCCC2)O)CCCCO1 c1(OC)cc(-n2nc(Cc3cccc(F)c3)nc2-c2ccc(F)nc2)cc(F)c1 CCCC(CCC)CC(=O)NCc1nc(C(N2CCC(C)(C(N)=O)C2)=O)co1 c1(NC(C=C2CC(N(CC(C3(C(N)=O)CC3)=O)CC3CCC3)C2)=O)nc(C)no1 N1(Cc2nnc(C(C)C)s2)CCS(=O)(=O)C(CCNC(c2conc2CN)=O)C1 N1(C(C2CC(C(C)C)C2)=O)CCN(C(=O)C=Cc2ncco2)C(CO)C1 C1(CCN(C(CCSCC(C)C)=O)C)CCN(C(=O)Cn2ccccc2=O)CC1 C1(CC)CCC(N=c2[nH]c(=NCC3CCOC3)[nH]c3ccccc23)CC1 c1(C(=O)NCCN(CCC)C(c2ccnn2C(C)C)=O)ncc(Br)cc1C C(CCC(C)(C)NC(C1(CC(C)C)CC(=O)C1)=O)NC(C(C)OC)=O CCCC(C)(CC)C(=O)N1CC(CNC(=O)CCCC2CC2)(OC)C1 C1(C(N2C(C)(CCO)CC2)=O)CCOCCN1C(C1CN2CCC1C2)=O C1(NC(c2ncsc2C2CC2)=O)CCCN(C(c2cc(-c3ccco3)no2)=O)C1 c1(NC(CC)CC)[nH]c(=NC2COc3cc(Cl)ccc32)nc2c1ncn2C CCC(C)N=c1[nH]c(=NC)[nH]c(=NCc2ccc(-c3nc[nH]n3)cc2)[nH]1 C(C)(C)(CCCC(=O)NCCN1CC2CC2C1)NC(c1ccc(CC)cc1)=O C1(C)(C(=O)NCC(C)NC(C2CC2C(F)F)=O)CCCCN1C(=O)OC(C)(C)C CC(C)(C)C(O)CC(N(C1(C)CCCC1O)Cc1cn(-c2ccc(Cl)cn2)nn1)=O N1(C(C(c2c(C)cccc2)(C)C)=O)CCC(CNC(=O)C(C)C)C(F)(F)CC1 N1(C(c2ccc(OC)c(Cl)c2)=O)CCC(NC(=O)C(C)=C2CC2)C(CO)CC1 c1(-c2cn(CC(=O)NCCCNC(=O)NC)nn2)ccc(C(C)C)cc1 c1(C(=O)NCC2N(C(C3CCC(C)CC3)=O)CCC2)nccc(N)c1Cl N1(C(C(CC)N(C)C)=O)CCC(C(=O)NCc2nc(O)ccc2C)=C(F)C1 CC1CC(NC(c2cccnc2C(F)(F)F)=O)CN1C(=O)CCCc1cncs1 C1(C(=O)Nc2cccc(NC(c3c(C)cn(C)c3)=O)c2)C2CC3CC(C2)CC1C3 CC(C)(CC(F)C(=O)N1C2C=CCC1CCC2)NC(C1CC=CC1)=O c1(C2CCN(C(c3ccc(C(C)(C)C(F)(F)F)cc3)=O)C2)ccc2c(c1)CCO2 c1(C(N(CCOC)CCNC(C2CCC(C(C)(C)O)CC2)=O)=O)cc(F)ccc1O Cc1cncc(C(=O)NCC2CCCC(CNC(C3CN(C4COC4)C3)=O)C2)n1 C#CCCCC(C)C(=O)N1CC2CCN(C(=O)CC(C)(C)C=C)C2C1 C1(Cn2c(CNc3cn(-c4sccc4)nc3)nnn2)CCCOCC1.C1CCCO1 N1(C(C2(F)CN(C(c3nn(CC)c(C)c3)=O)C2)=O)CCC(O)C(O)C1 C1(C(=O)NCC2C(C(=O)OCC)C2)C2CCC(C2)N1C(=O)C(C)N1CC(C)C1 c1(N2C3CN(C(C)=O)C(C3)C2)ccc(S(=O)(=O)NCC(O)C(C)C)cc1Cl C=CCCC(C(=O)OC)NC(=O)CC(CC1CC1)NC(=O)C1=NOCC1 C(=O)(CCCC(C)(F)F)NCC12CN(C(C3CN(CCC)C(=O)C3)=O)C(CC1)C2 N1(CC=C)CCC(C)C(C(=O)NCCCOC(=O)CCc2ccccc2OC)C1 CC(C)C(F)(F)CC(=O)NCC1(C)CN(C2CCN(C(=O)CNC(N)=O)CC2)C1=O Cc1ccc(F)cc1CC(N1CC(NC(=O)C(C)(C)C2CCC2)CC(O)C1)=O N1(C(C2CN(C(N(C)C)=O)C2)=O)CCCCC(NC(=O)CC2CCN(C)C2=O)C1 c1(C(N(CCN(C(CCOC)=O)C)C(C)C)=O)csc(-c2ccncc2)n1 c1(C(=O)NC(C)C2CC2)cc2ccc(-c3cccc(-c4nn[nH]n4)c3)cc2[nH]1 CCCCC(C)C(=O)N1CCN(C)C(C(=O)N(C)CC2(O)CCCC2)C1 CC(C)(C)C(=O)NCC(C1CCCC1)NC(c1cc(C(F)(F)F)n[nH]1)=O c1(C(=O)NC(CCNC(c2c(C)ccs2)=O)C(C)C)cccc(F)c1F C(CCC(C(=O)NCC1(C)CCC(C)CC1)NC(c1c[nH]ccc1=O)=O)OC CC1CN(C(c2ccc3c(c2)CCC3)C)CCc2ccc(F)cc21 CC(O)C(C(=O)NCC1CCCN1C(=O)C=CSc1nc[nH]n1)N(C)C C1(C(=O)NCC2(NC(C3=C(C)CCCC3)=O)CC2)CCc2nnc(O)n2C1 CC(C)CC(C(=O)N1CC2CN(C(c3cc(Cl)c[nH]3)=O)CCC12)C(C)C C1(N(C)C(C)C)CC2CCC(C1)N2C(C)N(c1cnc(-c2cccs2)o1)C(C)C CCC(CC(=O)NCCN(CC(C)O)C(C1CC2(C1)CC(C)C2)=O)C(F)F N1(C(c2c(CC)nco2)=O)CCCC2C1CCCN2C(=O)CN1CCCCCC1 c1(SC)cc(C(=O)NCC2(NC(=O)CC3CC3(C)C)CC2)ccc1N n1(CC(=O)NCCCCC(C)NC(=O)CC23CC(C2)C3)nc(O)ccc1=O c1(C(=O)NCCC(C)NC(C(CCCC)C)=O)cc2c(cc1OC)OCO2 N1(C(C(c2ccccc2F)C)=O)CC23CCCC2(CNC3)C1 C1(C(=O)NCC(CCC)NC(C2CC(O)(CN=[N+]=[N-])C2)=O)CN2CCN1CC2 C1(C(=O)NCCC(C)NC(Cn2c(C)ncc2)=O)CC12CCSCC2 c1(SCC2CC2CO)ccccc1Cl.c12cc(n[nH]1)NC2=O.C12CCCN1NC2 c1(C(=O)NCC(C)N(C)C(c2c[nH]nc2-c2ccccn2)=O)ccnn1C(F)F Cc1ccsc1CC(N1CCCC1C1(O)CN(C(=O)C(=O)NC(C)C)C1)=O C1(C(=O)OCC(=O)N(c2c(C)cccc2C)C2CC2)CC(N)CCS1(=O)=O N1(C(CSC)=O)CCC(C2(O)CN(C(=O)C(C)(O)C3CCC3)C2)CC1 C(CC(C(=O)N(CCN=[N+]=[N-])C)NC(c1cccc(CO)c1)=O)=CC CC(C)(O)C(F)C(=O)NC1CCC(NC(C2(CO)CCCC2)=O)C1 C1(CC=C)(NC(c2cc(Cl)c[nH]2)=O)CCCN(C(=O)C(CC)C(C)O)C1 c1(C(=O)NC(CC)(CNC(C2CC2(F)F)=O)CC)nn(C)c(N)c1C C1(N(C)C(C2CCNC(=O)C2)=O)CCC(NC(=O)CSCc2ccccc2)CC1 c1(CC)nn(C)c(CC(=O)NC2CCN(C(=O)CCCC#N)C(C)C2)c1Br c1(C(N(C)C)=O)ccc(C(=O)NC2CC(NC(c3ccc(F)s3)=O)C2)s1 c1(C(=O)NCC(CC)NC(c2c(N)cc(F)cc2F)=O)cnc2scc(C)n12 c1(C(=O)NC(c2cn(CC3CCOC3)nn2)C)sccc1F c1(OC)cc(C(=O)NC2CCN(C(=O)C=C(Cl)Cl)C(C)C2)cc([N+](=O)[O-])c1C c1(C(C)NC(c2ccns2)=O)nocc1C(=O)N(c1ccn(C(C)C)n1)C N1(C(c2ccc(SC)o2)=O)CCC2CCC(NC(C3(C)CC(C#N)C3)=O)C12 C1(C(=O)NCC(CC)NC(c2cc(C)cc(O)n2)=O)CC2OC(C)(C)OC2C1 CCCCC(C)C(=O)NC1CCCC(CNC(C2C3C4CCC(C4)C23)=O)C1 CC(C)(C)C(CNC(C1CC(=O)CCO1)=O)C(=O)N1CCC(CN=[N+]=[N-])C1 C=C(CC)CN=C(NCC1CCC1)NC1CCN(c2ccc(F)cc2)C1 C1(C(=O)NC2(C)CN(C(CCN(CCCCC)CCC)=O)C2)CC(C)OC(C)C1 C(CC1=CCCCCC1)NCc1[nH]nc(C(F)(F)F)n1 C(c1ccccc1Cl)=CC(=O)NC1C=CCN(C(C(CCC)O)=O)C1 N1(C(C2CCC3(CCC3)O2)C(=O)NC2CC(F)(F)C2)CCCCC1C1CCCO1 C1(C(N(C(C#C)C)CCCC)=O)CN(C(=O)CC2CC(=O)NC2=O)CC1C1CC1 C1(c2nnnn2Cc2ccccc2)(NCCC(CC)(C)C)CC2CC1CC2(F)F C=Cc1cnn(C)c1C(=O)NCCOC(C)(C)CNC(c1cnccn1)=O S(=O)(=O)(c1cccc(OC)c1)N1C(C(=O)NC(CCC)CO)CC1 c1(CC2N(CC(C=C)c3cccs3)CC2)cncc(F)c1 c1(OCCC(=O)NC2COCC2NC(C2C=CCC2)=O)ccc(F)c(F)c1 C(=O)(C(C)CC(F)(F)F)N(C(C)C)CCN(C)C(C1CCN(CCO)C(=O)C1)=O Cc1ccn(CC(=O)N(C)CC2(NC(c3cc(C(C)(C)C)n[nH]3)=O)CC2)c(=O)c1 c1(CC)ccoc1C(=O)NC(C(=O)NCCN1CCC(O)C1)c1ccoc1 Cc1cccc(C)c1C(=O)NCCC(O)CNC(C12CCC(C1)C2)=O C1(C(N(C)CC2(C)CCCO2)=O)N(C(=O)CCP(C)(C)=O)CCC1(C)C C1(NC(CC=CC=C)=O)CN(C(=O)Cn2nc(C)n(C)c2=O)CCC1C N1(C(CC=C)=O)CCN(C(=O)Cc2cc(C(F)(F)F)cc(Cl)n2)CC1CO c1(C(=O)NC2CC(CNC(CC3C(OC)CC3)=O)C2)c(C)cc(C)oc1=O C1(C(N2CCCC(NC(c3c(C)cc(O)nn3)=O)C2)=O)CCc2c(nnn2C)C1 c1(C(N(C(C)C)CCN(C)C(C2CC(=O)C2(C)C)=O)=O)c2c(nn1C)CCCC2 C1(O)(CNC(CCc2cc(C)[nH]n2)=O)CCN(C(c2cnn(C3CC3)c2C)=O)C1 N1(C(CCNC(C(C(C)C)N)=O)=O)Cc2ccccc2C(n2cccn2)C1 CCCCC(CC)CC(=O)N1CC(NC(c2cnc3ccsc3c2)=O)C1 Cc1ccc(F)c(C(=O)NC2(C3CN(C(c4cocn4)=O)C3)CC2)c1Br c1(C(=O)NC2CN(C(CC(C=C)CC)=O)CC2C)cccc(S(=O)(=O)NCC)c1 C1(CNC(C2C(C)=CCS2)=O)CN(C(C23CCCC(CO2)C3)=O)CCC12CCC2 N1(C(Cn2c(C)nc(C)n2)=O)CCCC(F)(CNC(=O)COC2CCCCC2)C1 c1(C(=O)NCC2C(CC)CN(C(=O)CC(C)(F)F)CC2)nc2ncccn2n1 c1(C(=O)NCC(CC(C)C)NC(CCCC(C)=O)=O)[nH]nc2c1COC2(C)C c1(CNC(=O)NCCNC(C2OCCC2F)=O)ccc(O)cc1F C=CCCN=C1NCCC(CSC)OC(=O)N2CCC(N1)C2.C(C)(C)(C)OC N(C1CCc2sc(Br)cc21)C(C)COCc1cccc(Cl)c1 C(=O)(C(O)C1=CCCCC1)N1CC(F)(C(N(C)CC)=O)C1 C1(C(=O)NCC2OCC3(CN(C(CC=CC)=O)C3)C2)CCc2nncn2CC1 C1(NC(C(F)=CCC)=O)CCN(C)C12CCCN(C(=O)C(C)(O)C1CC1)C2 C1(C(=O)NCCC2=CCN(C(C(CC)CC)=O)CC2)COc2ccccc2C1 CC(C)(CC(F)F)C(=O)NCC1CC(NC(c2ccccc2C(F)F)=O)C1 c1(CC)ccc(NC(=O)CCC23CC(CN2C(=O)C(C)(C)COC(C)=O)C3)cc1 N1(CCNC(C2C(NC(COCC(C)C)=O)CC2)=O)CCCOC1=O CCCCCCC(C)CC(=O)NC1C2CN(C(=O)COCC3CCC3)CC12 CC(O)C(F)(F)C(=O)NC1(CC(N)=O)CCN(C(C2CCOC2(C)C)=O)CC1 CC(C)CC(C)(CNC(=O)C(C)(F)c1ccccc1)NC(=O)COCCF n1(CC)cnnc1C(=O)NC1CCC(CNC(=O)CC2CSCCS2)C1 c1(C(C)(C)C)ccccc1C(=O)NCC1CN(C(C2CC23CC(O)C3)=O)CCO1 C1(C(=O)NCCCCNC(COC(C)=O)=O)CCCCC1F c1(C(=O)NC2CC(CNC(C3(SC)CC3)=O)C2)ccc(C)o1 N1(C(C(C)NS(CC)(=O)=O)=O)C2CCCC1CN(C(C1CCO1)=O)C2 c1(NC(=O)CSc2ccccc2)ccc([N+](=O)[O-])cn1 N1(Cc2cnc(C)s2)CC2CCN(C(=O)CCc3ncc[nH]3)C2C1 C#CCC(C)(C(=O)NOCC(F)F)NC(=O)Cc1c[nH]nc1C CCCCCC(C(=O)N1CC2CCCC1CN(C(=O)CC1(CO)CC1)C2)C(C)C CCC(C)(C)C(=O)C(=O)NCC(C)N(C(=O)C(C(=O)OC)C(C)C)C1CC1 c1(OC)ccc(C)c(C(=O)NCC(F)CNC(=O)C(C)(O)Cc2ccccc2)c1 n1(C2CCN(C(c3cc(C4CC4)n[nH]3)C(=O)NC)C2)ccccc1=O c1(CC(=O)NCCOCCCNC(CN2C(C)CC2)=O)nn(C)cc1Br C(CN(C)Cc1ccccc1)(C(=O)NCCCC1(O)CCC1)NC(C)=O c1(NC(=O)CC2(NS(=O)(=O)CCCl)CCC2)cnn(-c2ccccn2)c1 C1(CC(=O)NC2(C3CN(C(C(C)CN(C)C)=O)C3)CC2)CC2(CCC2)CCO1 C1(N2CCCC(C)CC2)CCN(C(=O)CC2CC3CCC2C3)CC12CC2 N1(C(C(C(=O)OCC)OC)=O)CCC(C(=O)NC(C)C(F)(F)F)C12CCC2 CCC(F)(F)CC(=O)NC(CC(N)=O)C(=O)N(C)CC1CCCC2CC12 Cc1nn(-c2ccncc2)cc1C(=O)NC1C=CCN(C(=O)CC2CC2(C)C)C1 C1(NC(c2ncccn2)=O)CCCC(C(N2CCCCC(CO)C2)=O)CC1 C(=O)(C(=O)CCC(C)C)N(CCC(N1CCC(N(C)C)C(C)C1)=O)CC=C Cc1nc(C)c(C(=O)NC(CNC(=O)C(C)(C)C2(C)CC2(F)F)CO)o1 c1(CCC(=O)Nc2ccccc2N2CCCC2)ccc(F)c(F)c1 c1(C(N(CCC(=O)NCCCc2nc[nH]n2)CC=C)=O)cc(O)ncn1 N1(C(c2cncc(N3CCCC3)n2)=O)CCN(C(=O)C=C2CCC2)C(CCO)C1 C(=O)(C1Cc2ccccc21)N1C(C(C)(C)NC(C(C=CC)O)=O)CCC1 c1(C(=O)NCC(C)(CO)NC(c2cc(O)ncn2)=O)cnc2n(c1=O)CCS2 C(=O)(C(CC1CC1)NC(=O)CNC(C1CCCO1)=O)NC.C12(CCCC1)CO2 N1(C(C2C(CC)CCCN2C(=O)C(OC)OC)=O)CCC2CN(C)CC2C1 O=C(CCCC(F)(F)F)NCC1CC(NC(c2cc3ccccn3n2)=O)C1 C1(C(=O)NC2CC(C)(CNC(C(CC=C)C)=O)C2)CC(S(C)(=O)=O)C1 N1(C(c2cccc(SC)c2)=O)CC2CC3CC2C1C3NC(=O)C=CCO N1(C(CC2CC(C(=O)OC)C2)=O)CCCC2(CCN(C(c3n[nH]cc3Cl)=O)C2)C1 c1(SCC(=O)NC(C(=O)OC)C)cccnc1.C12(CC1)CCCN(C(C)C)C2=O N1(C(COC(C)=O)=O)CCN(C(C2CNC(=O)C2)=O)C(C(C)C)C1 c1(C(=O)NCC2CN(C(C3CC(C4CCC4)C3)=O)CCO2)ccc2c(c1)OCO2 C1(O)(c2cn(CC(CC)(C)O)nn2)CCN(C(=O)Cc2cnccc2OC)C1 C1(C(N(C(C2CCC2)C)CC)=O)C2CC(O)C(C2)N1C(c1cccc(O)c1C)=O Cc1nc2ccccn2c1CC(=O)NCC1CCN(C(C2CC(F)C(=O)N2)=O)C1 N1(C(COCCOC)=O)CCC2(CC1)CC(C)N(C(c1cc([N+](=O)[O-])n[nH]1)=O)C2 C(c1cccnc1)=CCN(C(=O)CCCCN(C(=O)Cc1ccoc1)C)C C1(C#N)(C(N2C(C(N(CCOCC#C)C)=O)CCC2C(C)C)=O)CCCCC1 C1(NC(C=CC=CC)=O)CN(c2ncc(Br)cn2)CC(F)(F)C1 N1(C(=O)Cc2ccc(O)cn2)CCC(C2CN(C(C34CC5CC3C4C5)=O)C2)CC1 C1(C(C)NC(c2cn(C(F)F)cn2)=O)CN(C(c2cc(Cl)c[nH]2)=O)CCO1 Cn1c(C(N2CC(C)(NC(=O)CCN3CCC3)C2)=O)ccc1C#N N12CC(CCC1C)C2.c1(N(CCN(C(C)=O)CC)C(C)=O)ccsc1C c1(C(=O)NCC2N(C(C3CC(C)OC(C)C3)=O)CCCC2)cc(C#N)ccc1O C#CCC(CC#C)C(=O)NCCCC(C)NC(C1Cc2ccccc2O1)=O C1(C(=O)OC)CN(C(=O)CC(C(=O)O)N(C)CC2OCCN(C)C2)CCC1O c1(-c2cn(CC(=O)NCc3snc(C)n3)nn2)cnn(C)c1C c1(CC(N2C(CC)C(NC(=O)CN3CCC(F)CC3)CC2)=O)cc(F)cc(F)c1 N1(C(C(C)SCCCC)=O)CC2CC(C1)CN(C(=O)COCC(F)F)C2 CC(O)C(=O)N(CCC(=O)NC1CC(CCO)C1)CCCO C(=O)(C(C)CCCC(C)C)NCC1N(C(c2c(C)ccnc2)=O)CC(C)(C)C1 C=CCC(C(=O)NC(C)CCCO)NC(c1cnn(CCC)c1)=O c1(N(CC(=O)OC)C(=O)CN2CCOCC2CC(C)C)cc(OC)c(Br)c(OC)c1 C#Cc1cc(C(=O)NCC(C(C)(C)C)NC(=O)C(CC)CCOC)cc(F)c1 C1(OC(C)(C)C)CN(Cc2ccc(C3CCCC(=O)N3)cc2)CC12CC2 Cc1sc(Cl)nc1C(=O)NC(c1ccc(CNC(=O)C=Cc2ccsc2)cc1)C c1(C(=O)OC)cc(OC)cc(C(=O)NC2CN(C(=O)C=CC(C)(C)SC)CC2C)n1 c1(C(=O)NCC(CNC(C2(COC)CC2)=O)(C)OC)nn(C)c(C)c1Br CC(C)C(C)(O)C(=O)NCC1CC2CN(C(=O)Cc3ccc(O)c(Cl)c3)CC12 c1(N2CC=CC(NC(CS(CCC)(=O)=O)=O)C2)cc2c(cn1)C(=O)CCC2 N1(CCNC(C2C(C=C(C)C)C2(C)C)=O)CCCN(C(=O)CNS(N)(=O)=O)CC1 C(=O)(C(F)C(CC)CC)N1CC(C(C(=O)NCc2onc(CC)n2)O)C1 C1(CNC(c2n(CC)ncc2)=O)CC(C)(C)CCC1NC(C1(C)CCC1)=O c1(CC=C(C)C)ccccc1CC(=O)NC1CCCC1CNC(=O)Cc1ccsc1 CC1CN(C(=O)C=CCF)CC(C)N1C(C1CN(CC(F)F)C1)=O CC(C(=O)OC(C)(C)C)C(=O)N1CC(N(C)C(c2cc(C(C)(C)C)nn2C)=O)C1 C(=O)(C1COc2ccc(Cl)cc21)NC(C)CCNC(c1occ2c1CCOC2)=O C1(CC#C)CN(C(c2cnn(C(C)C)c2)=O)C12CCC2 c1(CC(N2C(CNC(c3cc(CC4CC4)on3)=O)CC2)=O)ccc(Cl)cc1 c1(C(C(=O)NCC(CNC(c2c(C)cco2)=O)O)C)ccc(Br)cc1F CCCC(CNC(=O)C(C)n1ccnn1)C(=O)NCCC(C)(C)C C(=O)(C1CCc2cccnc21)NCCCCNC(CC(C)(O)c1ccccc1)=O C1(CCC2N(C(C(F)=CCOC)=O)CCC2)CCCCN1C(=O)Cc1nc[nH]n1 C1(F)(CNC(c2c(C)nn(C)n2)=O)CCN(C(c2cnn(CCO)c2C)=O)CC1 c1(N(CCOCCCC)C)ncnc(NCc2cc(-c3ccco3)on2)c1C c1(C(=O)NCCN(C2CCCC2)C(CN2C(C)CC2)=O)c(F)c(F)cc(F)c1F C#Cc1cnc(C(=O)NC(CNC(C23CCOC(C)(C2)C3)=O)CC)c(C)c1 CCCS(=O)(=O)CC(=O)NCC1CN(C(c2cnc(O)cc2OC)=O)CC1C c1(C(N2CCOCC(CNC(C3CCC4CC34)=O)C2)=O)[nH]c2ccccc2c1Cl C1(C(N2C(CC(C)C)CC2)=O)CN(C(C2(N(C)C)CC2)=O)CC12CC2 C(CCC(=O)NC(C)C=CC(=O)NC(CC1CCCC1)CO)OCC CCC(F)(F)C(C)(C)C(=O)N1CCC(C2(NC(c3nc(C4CC4)cs3)=O)CC2)C1 C1(CNC(c2cnc(C(=O)OC)s2)=O)CN(C(c2ncc[nH]c2=O)=O)CC1(C)C c1(OCCCNC(c2cc(CCCC)n[nH]2)c2nnnn2C)ccc(Cl)cc1C c1(CC(=O)NCC2(NC(c3on(C)c(=O)c3)=O)CCCC2)nc2ccccc2s1 C1(CNC(C(C)OC)=O)C(C)CCCN1C(c1sccc1C)=O Cc1cc(=O)c(C(N2CCOC(C)C2C(=O)NCCCc2ncnn2C)=O)c[nH]1 C=C1COc2c(C(=O)NCCCNC(=O)Cn3cccc3)cnn2C1 C(=O)(N1OC2CC1C(O)C2O)C1CN(C(=O)C=CC2CCOC2)CC12CCC2 CC(CCC(=O)NC(c1nccs1)C)NC(=O)Cc1ccc(O)cc1 C=CCC(CC(=O)NCC(F)(F)Cl)NC(=O)CC(C)(C)C1CC1 C(=O)(C(=O)CC(C)CC)N(CC(N1CCCC(OCC#C)C1)=O)CCC C1(NC(C(C2CC2)OC)=O)CCSC12CN(C(c1ccc(F)c(C#N)c1)=O)C2 N1(CC)C(=O)CCCC1c1ccccc1.N(C(=NC)NCC)SC(F)(F)F C1(NC(NC(C#C)C(C)C)=NC(C)C)Cc2cccc(OC)c2C1 C1(C(N2CCC(N(C(=O)CCN3CCC3)CC)C2)=O)Cc2cc(F)cc(F)c2O1 Cc1ccc(F)cc1CC(=O)NC(CC1CCC1)C(=O)O CN1CCC(CCNC(=O)CCN(C)C(C2CCCCC2)=O)C1=O CC1CN(Cc2ccc(Cl)c(F)c2)CCC1CCC(=O)O N1(C(CC2CC(=C)C2)=O)CCN(C(=O)CCC23CCC(CC2)C3)CC12CCC2 N1(C(C)C)CC(NC(=O)NCC2(c3nn[nH]n3)CCCCC2)CC1=O CCC(CC(=O)N(C(C)C(=O)N1CCC1C(C)O)C)C(C)(C)C c1(C(N(CCCC(=O)NC(CC)(C)C2CC2)C)=O)cc(Cl)n(C)n1 c1(CC(=O)NC2(C)CCN(C(C(C=C)(F)F)=O)C2)cc(F)cc2c1OCOC2 C(CC(F)F)(C(=O)NCC1COCC1C(N)=O)N(C)C(c1ccc([N+](=O)[O-])o1)=O C1(CNC(CC=CCC)=O)CCN(C(=O)CN2CCCC2=O)CC1C1CC1 C1(CC(=O)NC(C(=O)NCCC2(C)N=N2)CC2CCC2)OCCC1(C)C C12(CNC(C(=O)NC(C)(C)CN3CCCC3)=O)CC(C1)C(Cc1ccccc1)O2 C(CC1=CCN(C(=O)CC2CC2C)CC1)NC(c1ccc(C(C)=O)cn1)=O c1(CN(CCNC(c2c[nH]c(=N)o2)=O)C(C23COCC2C3)=O)cccc(Cl)c1 C(=O)(CCC(=O)NC(C)CC(C)NC(C1(C)C=CCC1)=O)OC N1(C(CC=C)=O)CC(OCC)C(CNC(=O)CCc2n[nH]c(=N)s2)C1 Cc1cnc(C(=O)N(C)CCN(C(=O)CCCn2ccnc2C)C)c(Br)c1 n1(CC(N2CCC(C)C2CNC(C2CCCCS2)=O)=O)nc2ccccn2c1=O C1(CNC(c2ccncc2)=O)CN(C(=O)Cc2csnn2)CC1C(F)(F)F C(=O)(C(CC)C(=O)N1CCC(CO)(CNC(=O)CN2CCC(O)CC2)C1)OCC N1(C(C(C)(F)F)=O)CC2CN(C(c3ccc(F)cc3Br)=O)CC(C1)O2 C1(C)(C(=O)Nc2cc(CC)no2)CCCN1C(C1(c2cc[nH]n2)CC1)=O c1(C(=O)NC(C)C(C)(C)NC(C2CC23CCC3)=O)cnc2c(c1)NC(=O)CN2C c1(SCC)cccc(C(=O)NC2(C)CN(C(c3cccc(C(C)(F)F)c3)=O)C2)c1 c1(CCC)ccc(C(=O)NCCCN(CC(Cc2ccccc2)OC)CC)s1 c1(C(=O)NC(CN(C(c2coc(Cl)c2)=O)CC)C)cn(C(F)F)nc1C(F)F N1(C(c2nn(CC)c(C)c2)=O)CCC2(CC2C(=O)Nc2cccc(C3CC3)n2)C1 CCC(C)C(=O)C(=O)N1CCOCC(NC(C2C=CCS2)=O)C1 Cc1nn(C)cc1-c1ccc(C(=O)N(C(C)CCO)Cc2ccccc2)nc1 C=C(C)CC(C(=O)OC)NC(C1CCCCN1C(c1cnc(O)n1CC)=O)=O c1(C(N(CCNC(C2C(CC)C2)=O)CCOCCO)=O)snc(O)c1Cl N#Cc1cc(C(=O)NCC2(O)CC(C(=O)NCCC34CC(CO3)C4)C2)c[nH]1 CCCCCC(C(=O)NC1CCCC1NC(c1ccnn(C)c1=O)=O)C(C)C c1(NC(=O)Nc2cccc(C(C)(F)F)n2)cn2ccc(Br)cc2n1 N1(C(COCC(=O)NC)=O)CCC(C(=O)NC(COC)CC)(C(C)C)C1 CCC(C)C(C(=O)Nc1ccc(F)cc1C)N(CC)Cc1cnn(C)c1 CC(CNC(=O)CNC(=O)CC1CCC=CCC1)C(F)(F)F c1(C(=O)NCC2(O)CN(Cc3ccccc3)C2)ccc(I)cc1Br C1(C(=O)NC(c2cccnc2N2CCCC2)C2CC2)CC2(C1)CC(F)(F)C2 C(CNC(=O)CCc1cncc(F)c1)(C(C)C(C)C)NC(C1(COC)COC1)=O c1(C(N2CCC(CNC(COC(CC)CC)=O)C2)=O)ccc2nc(O)oc2c1 CN1CC(C)(C)CC1C(=O)NCCCCCCNC(=O)CC=C(Cl)Cl Cc1nc(C(=O)NCC2COC(CNC(c3c[nH]c(C(F)(F)F)c3)=O)C2)nn1C C1(CC=C)(NC(=O)Cc2nc[nH]n2)CCCN(C(=O)C=C2CCCCC2(C)C)C1 c1(OC)cc(C(N2CCC(c3ccon3)C2)C(=O)NCCCC2CC2)sn1 N1(C(C23CC(NC(C4C(COC)CC4)=O)(C2)C3)=O)CCCNC(=O)CC1 n1(C(C)C)cnc(C(=O)NCC(CO)NC(=O)C(C)(C)c2cccs2)n1 c1(NC(C=CCN(C(=O)CC2CCCC(O)C2)C)=O)cccn2nccc12 c1(NCC(C(=O)OC)(F)F)ncc2ccc(-c3ccnc(Cl)c3F)cc2n1 N1(C(CNC(C2C(C)C2)=O)=O)CC(C)(C(N2CC3(CCC3(C)C)C2)=O)CC1(C)C Cc1cccc(C)c1C(=O)NC1C=CC(CC(N2CC3(CCN3C)C2)=O)C1 N1(C(C(C(C)C)(C)C)=O)CC23CCCCC2(C1)CN(C(C1CCC(C)CC1)=O)C3 C1(C(N2CCC(NC(C(CC)SC)=O)(CF)C2)=O)Nc2ccccc2C1(C)C N1(C(CCNS(C)(=O)=O)=O)CCN(C(c2cc(Cl)ccc2F)=O)C(CF)C1 C12(CNC(C=CC(C)C)=O)CC1CN(C(C1(O)CC(C(=O)OC(C)(C)C)C1)=O)C2 C1(NC(c2[nH]cc3c2CCC3)=O)CCN(C(=O)CC2CCCO2)CC1F c1(CNC(c2ccc(C(F)(F)F)c(Cl)c2Cl)=O)cccc2ncccc12 c1(C(C2CC2)NC(c2nnc(N(C3CCN(CCC)C3)C)s2)=O)ccc(NC)cn1 N1(C(C2CCCCC23OCCO3)C(=O)NCCOC)CCC2(CCCCCC2)C1 c1(C(=O)NCC2C=CC(NC(C(C(C)C)NC=O)=O)C2)noc2ncccc12 c1(C(C)C)c[nH]cc1C(=O)NC(C(=O)NCCN1CCC(C)C1)c1ccco1 C1(C(=O)NCC=CCCOC)CC=CC(NC(C2CCOC2C)=O)C1 C1(NC(C(C)OC)=O)CC2CC1N(C(C1CCN(OC)CC1)=O)C2 CC1CC(NC(=O)CCn2cnc(=N)[nH]2)CCN1C(=O)Cn1nccn1 C1(NC(C2CC(SC)C2)=O)CCC2(CC1)CC2NC(c1cccc2nccn12)=O Cc1c(I)cc(CN2CC(C)CC2C(=O)Nc2cccc(F)c2[N+](=O)[O-])cc1I CCCCC(CC)CC(=O)N1CCCC(NC(c2nnn(C)c2C)=O)C1C N1(C(CC2CC(OCC)C2)=O)CC(C)CN(C(c2nc(Cl)cs2)=O)C(C)C1 C1(C(N2CC(C3(Cc4cccc(C)c4)CC3)C2)=O)CCc2nc(C)cn2C1 c1(OC)ccc2c(C(=O)NC(C)CCNC(c3cccn3C(C)C)=O)n[nH]c2c1 N1(C(C(C#N)CC2CC2)=O)CC=C(C(=O)N2CCCN(CCO)CC2)C1 C1(CC)CCCC(C(N2CCC(N3CC(C(=O)OC(C)(C)C)C3)C2)=O)O1 C1(NC(c2c(CC)csc2)=O)(CO)CCN(C(=O)C(CC)C2CCOCC2)C1 c1(C(=O)NC(CNC(C2CC(C)(C)O2)=O)CO)c(Cl)ccc(Br)c1F c1(OC)cccc(C(C)C(=O)NCCCNC(=O)CC2CC3CC3C2)c1 Cc1oc2cc(C(=O)N(C3CCN(C(=O)C=CC(C)(C)C)C3)C)[nH]c2c1C CCC(CO)(CO)C(=O)NCc1c(C(F)(F)F)coc1C C1(C(=O)NCC2CC(C(=O)NCC(CC)(C)OC)C2)CC2(CC2)CO1 c12cc(cnc1OC)C(=O)N2.C1(SC)COCCN1C(=O)NCC1CCCCC1 Cc1cc(C(=O)NCCC(C)N(C)C(C2CC(C)C2)=O)c2c(n1)CCCC2 c1(C(=O)NCCC(CNC(C(C2CC2)OCC)=O)O)cc(C(F)(F)F)cc(O)c1 CC1(CO)CCCN1C(=O)C(C1CCN(C(c2cccc(O)c2)=O)C1)F C12(CNC(c3c(OC)csc3)=O)CC1CN(C(=O)C(C)Oc1ccc(F)cc1)C2 C1(CNC(C2(OC)CCSC2)=O)COCCN1C(c1ccn(C2CC2)n1)=O C(=O)(C(C)CCCC(C)=O)NCc1ccc(C(=O)NC(CC)C)cc1 c1(C(=O)NC(C(=O)NCCC2CN(C)C(=O)C2)CCF)cc2cccn2cn1 Cn1ncc(Cl)c1C(=O)NCCC(C)(C)NC(=O)CCC1CCC1 C1(NC(=O)Cc2cc[nH]n2)CCN(C(C2(Cc3cnn[nH]3)CCC2)=O)CC1O c1(C(=O)NCCCN(C(c2nn(C)nc2Br)=O)CC)ccc(Cl)cn1 C1(c2n(CCCOC)nnn2)(NC(c2sc(C)nc2C)C)CCCSC1 C1(NC(C(C)(C)C)=O)CN(C(c2cc(-c3ccccc3F)on2)=O)CC1O CCCCCCCCC(=O)NCCCCC(C)NC(=O)C(C)n1ccnc1 C1(C(=O)NCc2cn(CCNC(C3CCC(C)O3)=O)nn2)CCCC2(CCC2)C1 CC1(C)C(CNC(C2CC23CCC3)=O)CCN1C(=O)CN1OC(C)(C)CC1=O c1(CN)cc(F)nc(O)c1Cl.C12CCCCN1C(=O)C(=O)N1CCC2CC1 c1(CC)cnc(O)c(C(=O)NC2(CNC(c3cnn(C)n3)=O)CCCCCC2)c1 C1(NC(c2cccc(CCO)c2)=O)CN(C(C2CCSC2)=O)CC(F)(F)C1 c1(C(=O)NC(CN(C(c2cnn(CCF)c2)=O)CC)C)ccn(C)c1C N1(C(c2nc(N(C)C)oc2)=O)CC(CO)C2(C1)CN(c1nnc(C(F)F)o1)C2 C(CC(CC)C(=O)N1CC2CC(NC(=O)Cc3cc(C4CC4)nn3C)C1C2)=CC C1(N(C(C2C(OCC)C2)=O)C)CCC(NC(=O)Cc2ccccc2C(N)=O)CC1 c1(C(C)C)cc(C(N2CC=CC2CNC(=O)CC(O)CN(C)C)=O)nn1C c1(NC(N2CCC(NC(C(C=C)C)=O)C2)=O)sc2c(c1C#N)CCCCC2 N1(C(CCOCC)=O)CCN(C(C2(CC(C)C)CC2)=O)CC12CC2 S(=O)(=O)(c1ccc(F)c(Cl)c1)N1C2C(C(=O)NCCC)C(C2)C1 C1(C(N2CCC(NC(=O)Nc3ccc(O)cc3)CC2)=O)CCCC2(CCC2)C1 CCC(C(=O)NCC(O)CNC(=O)Cc1ccc(CO)cc1)C(C)(F)F c1(NC(C2(C)CCCN(C(c3cocn3)=O)C2)=O)ccc(Br)c2ccccc12 N1(C(C(C)NC(N)=O)=O)CC2CCC1CN2C(c1cscc1C(F)(F)F)=O c1(OCC(=O)NCC2COCCN2C(c2cc(Br)c[nH]2)=O)cncc(Cl)n1 C(C(C(C)C)NC(=O)C(C)(F)F)(c1ccccc1)NC(c1[nH]cc(CC)c1)=O c1(OCCNC(N(CCCC)Cc2cccs2)=O)ccc(C)cc1 N1(C(C=CCCC(C)C)=O)CCSCC1C(=O)N(CCC(C)(C)O)C N#CC1CN(C(c2nc(C(=O)N(c3ccc(Br)cc3CO)CCO)cs2)=O)CCO1 C1(N(C(C2SCC=C2C)=O)CC)CCN(C(C2CN(C(C)C)C2)=O)CC1 C1(C#CC(=O)N2CCCCC2C(C)(C)CNC(=O)C(=O)NC(C)C)(CC)CC1 n1(C(C)C(=O)N(C2CN(C(C3CC4CC4C3)=O)C2)C)ccc2ccccc2c1=O N12CCCC1C1(CC1)C2=O.n1(CNC(C2CC2CF)=O)cc(CO)nn1 C(CCCCCCO)NC(C1C(CNC(C2CC(CF)C2)=O)CCC1)=O c1(OCC(=O)N(C2CN(C(=O)NCCOC)C2)C)ccc(SC)cc1 C1(C2CCOCC2)(C(=O)NCC2C(C)CCN(C(c3c(C)nccn3)=O)C2)CC1 CC1OC2(C(N3CCC(CNC(=O)CCN4CCOCC4)C3)=O)CC1C2 c1(C(N2CCC(COC)(NC(=O)Cn3cncn3)C2)=O)ccc2scnc2c1 CC1=C(C(=O)NC2(C3CN(C(=O)C(c4ccc(C)cc4)O)C3)CC2)CCC1 N1(CC)CCC(C(=O)NC2CC(CNC(c3csc(Br)n3)=O)C2)C1 c1(C(=O)NC2C(CNC(C(C(C)(C)C)N(C)C)=O)C2)c(Br)ccc(F)c1N c1(C(N(C2CCN(C(c3cccc(Br)c3N(C)C)=O)C2)C)=O)cc(I)cnc1Cl c1(C(=O)NC2CC(CNC(Cc3scc(C)c3)=O)CC2O)ccc2cnoc2c1 CC(C)P(=O)(CC(=O)NCC1(O)CCN(C(=O)Cc2c[nH]ccc2=O)C1)C(C)C Cc1cc(C(=O)NC2CC(NC(c3ccccc3)CCO)C2)c(C)[nH]1 C(=O)(C(F)(F)C(F)(F)C(F)F)N1CC(C2CN(C(c3n(C)c(C#N)cc3)=O)C2)C1 c1(OC)n[nH]cc1C(=O)N(C(C)CCNC(=O)C(F)(F)c1csc(C)c1)C c1(C(=O)NCC2CCC(C)CN2C(C2CCSCC2)=O)cnc2[nH]cncc1-2 c1(C(=O)NCCCC2N(C(C(C(C)C)C)=O)CCCC2)cc2n(n1)CCCC2 N1(C(C(C)n2ccnc2)=O)CC(CNC(C2CCN(CC3CC3)CC2)=O)C(O)C1 O=C1CCC2CN(c3cc(NCC4CCN(CC(F)F)CC4)ncn3)CCC2N1 C(=O)(C1=Cc2ccccc2OC1)N1C2CC(NC(=O)C=CC(F)(F)F)CC1CC2 c1(C(=O)NC(C)CCNC(c2cccc(CN=[N+]=[N-])c2)=O)cc(F)c(F)cc1N c1(C(=O)NC2CC(O)(CNC(C(CSC)O)=O)C2)cccc2sncc12 C12(NC(CS(C)(=O)=O)=O)COCCC1CN(C(c1cnc3[nH]cnc3c1)=O)C2 n1(COC)nccc1C(=O)NC1CC1CNC(=O)COC1(C)CCCC1 C12(C(=O)NCc3ccc(C(N(C4C(C)CC4)C)=O)o3)CCCC1C2(F)F c1(C(=O)NCC2CN(C(Cc3cc(C)sc3C)=O)C(C)C2)cc(C)n(C)c(=O)c1 N1(C(c2c(C(C)=O)ccs2)=O)C2CCC1CC(N(C(=O)Cc1c[nH]nc1C)C)C2 c1(C(=O)NCC2C(CNC(C3(C(=O)NC)CCC3)=O)C2)coc2ccc(Cl)cc12 C(=O)(C(C)(O)CC(C)C)NC(CC)CN(C)C(C1(N(C)C)CCC1)=O N1(CC(=O)NS(CC)(=O)=O)CCS(=O)(=O)C(CCNC(=O)CC(C)(F)F)C1 c1(C(=O)NC2CC(F)(CNC(CC3(C)OCCO3)=O)C2)ccc(N=S(C)(C)=O)s1 C1(CNC(CC2C(C)(C)CC2)=O)CC2CCC1N2C(=O)Cc1sc(O)nc1O c1(-c2ccc(C)nc2C)ccc2c(c1)COC21CN(Cc2cc(F)cc(Br)c2)C1 Cc1cc(C(=O)NC(C)C(C(C)C)NC(=O)CN(C)C2CC2)n(C(C)(C)C)n1 C1(O)(CN(C)C(c2conc2C(C)(C)C)=O)CCN(C(=O)C(C)(C)CC2CC2)C1 Cc1ccncc1CC(N1CCCC1C1(NC(=O)CC2CC2C)CC1)=O O=C(C#CC1CCCCO1)N1CCC2CN(C(C34CCCC(CO3)C4)=O)CC12 C=CC(C)(CCOC)C(=O)NC1CCN(C(=O)CNC(C2CCOCC2)=O)C1 N1(C(CCCN(C(C)=O)C)=O)CCCC(CN(C(=O)CC2CC3CCC2O3)C)C1 Cc1cc(C)c(C(N2CC3(CCC3)CC2CNC(C2CC2(Cl)Cl)=O)=O)c(O)n1 N1(C(C(C)C)=O)CCCCC1C(=O)N(C)CCN(C(=O)Cc1cccc(F)c1)C C1(C(N(CC(CNC(C2(OC)CCOC2)=O)O)C)=O)CCCCCCC1 N1(C(=O)CN2CC=CC2)CC2(CO)CC1(C(=O)NCC1(C3CC3)CCCO1)C2 c1(C(N2CC(NC(CC3(C(=C)F)CCC3)=O)C(SC)C2)=O)cnc2sccn12 c1(OC)ccc(C=CC(=O)N(C2CN(C(=O)C(C)CS(C)=O)C2)C)c(C)c1 N1(C(CC(=O)OC(C)(C)C)=O)CC(NC(C2CCCC2CF)=O)C2(CC2)C1 CCCC(C)(O)CC(=O)NC1CCCCN(C(c2ccc(F)cc2F)=O)C1 N1(C(C2(c3nn[nH]n3)CC(C)C2)=O)CCCC(C#N)C1 c1(CCC(=O)NC2(COC)CN(C(=O)CCC3(C)N=N3)C2)nc2ccccc2[nH]1 C1(C)(NC(=O)NCC(c2ccccc2)(C)C)CC(CO)C1 CC(C)C(O)C(F)(F)C(=O)N1CCCN(C(=O)CCCCN2CCOCC2)C(C)C1 C(=O)(C1CCc2ccccc21)NCC1C(C(=O)NC2C(C)N3CCC2CC3)C1 C12CCCC(C1)C(=O)NCC(C)(C)NC(=O)N2.C1(O)(C(=O)NNCC)CCC1.CC C1(CCNC(C23CC(F)(C2)C3)=O)(OC)CN(C(=O)CCC2CC2(Cl)Cl)C1 N1(N(C(c2nc(Br)sc2Cl)=O)CCN2CCOCC2)CCCC(C2CCCCC2)C1 Cn1cc(C(=O)NCCC2CCN(C(C3(CO)CCCO3)=O)C2)c(O)nc1=O N1(C(C23OCC(C)(C2)C3)=O)CC2CCC(C1)N2C(C1(C)CC(F)(F)C1)=O C=CCCCCCCCC(=O)NC12COC(C1)C(NC(=O)CCN=c1[nH]ccs1)C2 C1(C(=O)NCC23OCC(NC(=O)CCc4nccs4)(C2)C3)COC2COCC12 c1(C(=O)Nc2c(C)cc(O)nc2)cnc2c([N+](=O)[O-])cnn2c1 c1(C(N2CCC(C)(C(=O)NC(C(=O)OCC)C3CC3)C2)=O)cc2ccccc2o1 C1(CNC(=O)CC23CCCC2C3)CC2CN(C(c3csc(F)c3)=O)CC12 CC1(CNC(c2ccc(NC(N)=O)cc2)=O)CCCN1C(=O)COC(F)F c1(CNC(CC2CN(C(C=CC=CC)=O)C2)=O)cc2cc(Br)ccc2s1 c1(C(N(CCC)CCNC(c2nc(C(C)C)oc2C)=O)=O)cc2cnccc2o1 C1(CNC(=NC)NCC2(C3CCC3)CC2)CCCCC1C1CC1 S(=O)(=O)(c1ccccc1)N1CC2C(CNC(c3cnnc(Cl)c3)=O)(C2)C1 C=CCCCC(C1CC1)NC(c1cn(CCNC(C2(C)CC(F)(F)C2)=O)cn1)=O c1(C(=O)NC2C(NC(C(CCC)C)=O)C2)c(CC)cccc1F c1(OC)ccc(CO)cc1C(=O)N(C(CNC(=O)CC1(O)CCCC1)C1CC1)C N1(C(C(C)SC(F)(F)F)=O)CCC(C)(C(=O)NCCn2ncccc2=O)C1 Cc1cc2ccc(C(=O)NC3CN(C(=O)C4=CS(=O)(=O)CCC4)CC3O)cc2o1 c1(CNCCCC)nc(CN(CCC)C(c2ccco2)C)no1 N1(C(C2CC(C)(C(C)(C)C)C2)=O)CCC(NC(c2csc3nccn23)=O)C12CC2 N1(C(c2nc(C)sc2)=O)C2CCC1CC(CNC(c1ccnnc1Cl)=O)C2 N1(C(C=COCC)=O)CCC2(CCCC2NC(c2cc(C3CC3)ncn2)=O)C1 C1(C(N(C2C(C)CCC2)C)=O)CC2CN(C(C3(C)CCOCC3)=O)CC2C1 C=C(C)C1CCC(C)=CC1CC(N1CCC(C)(NC(=O)CC2CC(C)C2)CC1)=O C1(CC(=O)NCC2CN(C(c3nc(C)sc3)=O)CC2(C)C)CCn2cncc2C1 C1(CC)CN(C(=O)CC2CCCCC2O)CC1NC(C1(CO)CCCO1)=O C(c1ccc(F)cc1)=CC(=O)NC1C(NC(CN(C(C)=O)C)=O)C1 CC(c1ccccc1)=CC(=O)N(CCC(C(C)(C)C)NC(c1sccc1C)=O)C C1(C(N)=O)CN(C(C2CCN(C3CC3)CC2)=O)CCC1NC(c1ccsc1)=O Cc1nc(CCN(C(=O)C(C)N(C(=O)CNc2ccccn2)C)C)no1 C1(NC(C2C3CCCC23)=O)CCSC12CN(C(=O)CCCN1CCCC1)C2 Cc1cn2c(n1)CC(C(N1CC(C(C)NC(c3cc(Cl)sc3Cl)=O)C1)=O)CC2 Cc1ncc(C(=O)N(C)CC2CCCN2C(c2ccc(O)c(F)c2)=O)c(O)n1 C1(C(N(CC(C)(C)NC(=O)C(F)=C2CCCC2)C)=O)CC(C(F)(F)F)CO1 N1(C(CCCOC(C)=O)=O)CCSCC1C(=O)N(C(C)CCN(C)C)C c1(CNC(C23N(C(=O)CC45CCCC4C5)CCC2C3)=O)ccc(F)c(F)c1 C1(NC(CC(CC)O)=O)CC2CCC(C1C)N2c1nnc(C(F)F)s1 C1(NC(=O)CCc2ccccc2)C2CCN(C(=O)C=C3CCSCC3)CCC12 Cc1coc(C(C)C)c1C(N1CC(NC(C23CCC2C3)=O)C(F)C1)=O c1(C(=O)NC2CCC(NC(C3(Cl)CC34CCC4)=O)C2)c(Cl)ccc(F)c1F Cc1nncn1CCCNC(=O)NCC1CCCCS1 C(C)(C)(CC(C(=O)NCc1ccc(F)cc1)N(CCCF)C1CC1)SC c1(C(C)=O)ccc(C(=O)NC2CCCCC2CNC(=O)CCNC(=O)CO)nn1 N1(S(c2cccc(C#N)c2Cl)(=O)=O)CCc2nc(C3=CCC(O)CC3)sc2C1 C(C(=O)NC(C)(C)CCNC(C1CC=CCC1)=O)(C(C)C)NC(CC(C)C)=O c1(N2CCC(N(C(C(COC)O)=O)C)C2)ncnc2ccc(O)cc12 Cc1c(C(=O)NC2CCN(C(C3CC(F)(F)C3)=O)C(C)C2)nn2ccccc12 c1(N2CCC(CC(C)NC(C3(CCC)CC3)=O)CC2)c(F)cccc1[N+](=O)[O-] C(=O)(C(=O)CC(C)CC)N(CCCNC(C(C=C)CC)=O)CC c1(C(=O)NC(CCCC)CNC(=O)CSCCCC)ccc(OC)c(Cl)c1F N1(C(c2cc(CC)nn2C)=O)CCOCC(NC(C2(F)CC=CC2)=O)C1 C1(CNC(C2CN(C(C)=O)C2)=O)CCCN(C(C2NC(=O)OC2C)=O)CC1 c1(C(=O)NCCN(C(C)C)C(C2C=CC=CC=C2)=O)cc2n(n1)CCOC2 c1(C(N2CCC(COC(C)=O)C2)C(=O)NCC(C)C)ccc(C(C)C)cc1F c1(SC(C)C(=O)Nc2cc(Cl)ccc2-n2cncn2)ccc(Br)c(Cl)c1 CCCC(O)CC(=O)NCC1(CNC(C2CC23CCOCC3)=O)CC1 N1(C(CC(C)OC)=O)CCCC(C)(CNC(=O)C=Cc2ccco2)C1 S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1C2CC(C(N3CCC(F)(F)CC3)=O)C1CC2 C1(C(c2ccccc2)OC)C(O)C(O)CCN1C(=O)C(C)(C)CC(F)F C(=O)(C(CNC(=O)C(C)S(N)(=O)=O)(CC)CC)N1CCN(C(C#C)C)CC1 C(c1cccc([N+](=O)[O-])c1)=CC(=O)NCCN(CC1CC1)Cc1ncccc1Br C#CC1(C=C)COCCN1C(c1n[nH]cc1C(F)(F)F)=O c1(OC)ccc(=NC(=O)CC2CCCCCCC2)[nH]c1C(C)=O C1(NC(=O)CCc2ncccn2)C2CN(C(=O)CCc3nc[nH]n3)CC12 N1(C(c2c(C)csc2)=O)CCCC(C)C1CNC(C1(C)CCC(F)(F)C1)=O Cc1ccc(NC(=O)C(N2CCC(NC(F)(F)C(F)(F)F)C(C)C2)=O)c(C)c1 c1(-c2ccc(C#N)nc2)cccc2c1CCN(S(=O)(=O)CC1CCCC1)C2 C1(NC(C(C)(C)NC(=O)NCCC)=O)CN(C(c2cccc(=O)o2)=O)CC1C CCC(O)C(C)C(=O)NCCNC(C1CCCN(C(=O)Cn2ncnn2)C1)=O C1(C(=O)NC2CCC(CNC(c3ncccn3)=O)CC2)CCC=CCCC1 C1(C(C(=O)NCC(C)N(C)C(C2(C(F)(F)F)CC(O)C2)=O)OC)CCCCCC1 c1(C(N(CC(CNC(C(CC)CCOC)=O)O)C)=O)cc2c(s1)CN(C)CC2 C1(CCC)CN(C(C2(CC)CC2(F)F)=O)CCN1C(=O)CC1CCCCCC1 N1(C(c2c(CCC)cccc2)=O)CC2CCOC2(CNC(c2nn[nH]c2Cl)=O)C1 c1(C(N2CC(CNC(c3c(C)cc(CC)o3)=O)OCC2)=O)ccc(F)c(SC)c1 CN1CCC(F)(CNC(C2(C(=O)NC3CC4(C(C(=O)C5CC5)C4)C3)CC2)=O)C1 C12(NC(c3nc[nH]n3)=O)CCC(C(=O)Nc3ccc(Cl)cc3I)(CC1)CC2 C(Cn1ccnn1)(C(=O)N1CCC(C(OC)OC)C1)N(C(C)(C#N)C1CC1)C N1(C(CCC(C)C)=O)CCCN(CC2CC3(C)CC2CO3)CC1c1ccccc1 C1(CC)CCCN(C(c2ccc(OC)o2)=O)C1C(=O)NCCCCC1CC1 C12CCN(C(=O)O)C(C)C1C2.N1(CCOC)CCN(C(C(C)(C)C)=O)CC1 c1(C(=O)NCC2(O)CN(C(C34CC(OC)C3C4)=O)C2)cccc2c1CCCC2 C1(n2ccnn2)CCCCC1SC.C1(C(=O)NCCSCC)CC1C(=O)O.CCS N1(C(C2(CC#C)CCC2)=O)CCCC(NC(=O)CC(C2(OC)CCCC2)C)C1 N1(C(c2ccc(F)cc2Cl)=O)CCC2(CCCCN(C(C34CSCC3C4)=O)C2)C1 c1(C(N2CCC(NC(C3(COC)CC3)=O)C2)=O)cc(Br)cc2c1OCO2 C1(C(N2CCN(C)CC2CNC(=O)CC(F)(F)Cl)=O)CCc2[nH]nc(O)c2C1 C=C(C)CC(C)C(=O)N1CCCCC1C1CCN(C(=O)CCCOCCC)CC1 CC1=C(C(=O)N2CCC2CNC(c2ccc3oc(C)nc3c2)=O)C(=O)OC1(C)C C(=O)(C(C)(C)C(=O)N1CCN(C)C(CNC(c2nc(=O)n(C)[nH]2)=O)C1)N(C)C CCC(CC(=O)NC1CCN(C(=O)C=C(C)c2cccc(Cl)c2)CC1)C(C)(C)C C1(F)(C(=O)NC2C(CNC(CSCC=C)=O)CC2)CC2(CCC2)C1 N#Cc1ccnc(C(N2CC3C(CNC(=O)C=CCF)C3C2)=O)c1 Cc1nc(C(=O)NC(CNC(=O)CC2CCN(C)C2=O)C(C)(C)C)cn(C)c1=O N1(C(COC)C)CCCC(C2CCCN(C(c3cc(C)nn3C)=O)C2)C1 C1(C(=O)NC(CC=CC)C(=O)N(C2CC2C)C)CCC(O)CN1C C(=O)(CC1CC(O)c2ccccc21)N1CCN(C(C(C)=C2CC2)=O)C(C)C1 N1(C(COC(CC)C)=O)CCCC1(C)C(N1CCC1CF)=O NS(=O)(=O)c1cccc(C(=O)NCC2CCCN(C(c3cn[nH]c3)=O)CC2)c1 Cc1nn(C)c(NC(C2CC(C(=O)NCc3sccc3Cl)C2)=O)c1Br n1(CC(=O)NCC2N(Cc3occ(C(=O)OCC)c3)CCC2)ncn(C)c1=O C(=O)(C(CP(C)(C)=O)C(F)(F)F)NC(c1ccc(OC)cc1)C1CC1 N1(C(c2cncc(OC)c2)=O)CCCC(NC(=O)C=CC2CCCCCC2)C1C CCC(CNC(C1Cc2nccn2C1)=O)(CC)C(=O)N(C1CC(SC)C1)C Cc1cccc(CN2CCC(O)C2C(=O)Nc2ccc(Cl)c(F)c2)c1O N1(C(C(n2ccc(C)n2)C)=O)CC(NC(=O)C(S(C)(=O)=O)C2CC2)C(N=[N+]=[N-])C1 c1(CC)nccnc1C(=O)OC.C12CN(CC1C)C(CCNC(C)=O)C(=O)N2 c1(NC(c2ccc(OCCC)c(OC)c2)=O)cc(Br)c([N+](=O)[O-])cn1 c1(OC)cc(N2CC3(CC3)CC2CNc2ccccc2SC)nc(S(C)(=O)=O)n1 N1(S(CCOC)(=O)=O)CCn2cc(C(N3CC4(CCOC4)C3)=O)nc2C1 CC12CN(C(=O)CCS(C)(=O)=O)CC1CN(C(c1n[nH]c3c1CCC3)=O)C2 N1(C(c2c(C)snn2)=O)CC2CC(C(=O)NC3(C4CC4)CCCC3)(C2)C1 C1(NC(CN(C)C(=O)C2CC2)=O)COCCC1NC(C1(CF)CC1(F)F)=O c1(CCC(=O)NC(C)C(C)(C)NC(C2CC2C)=O)csc2nc(C3CC3)cn12 C1(N(C(c2cc(F)ccc2OC)=O)CC)CCCN(C(=O)OC(C)(C)C)C1C Cc1ncc(NCc2nncn2CC(F)(F)F)c(C#N)n1 c1(C(CO)NC(C2C=CC(NCc3ccnc(Br)c3F)C2)=O)ccc(F)cc1F C#CC1COCCC1N1CCN(C(=O)Cc2cnn(CC)c2)CC1 C(C)(C)(CCCNC(C1(C#N)CC1C(F)(F)F)=O)NC(C1C(CC)C1)=O C1(CC(N2CCC(CC)C2)=O)C2CCCC2N1C(c1cc(OC)ccn1)=O c1(CC)ccccc1C(F)(F)C(=O)NC(C)(C)C(C)NC(=O)C(C)n1ccnc1 C(C(CC(F)(F)F)NC(C12CCC(C1)C2(C)C)=O)NC(C=C1CCN(C)C1)=O N1(C(CCCCSC)=O)CCC(N(C)C(c2ccnc(CO)c2)=O)C(C)C1 c1(OCCOC)ncccc1C(=O)NCC1CCN(C(=O)C(F)C2CCC2)C1 c1(-n2cc(C(=O)NC3CCN(CC4(F)CCCCC4)C3)nn2)ccc(CO)cc1 c1(C(=O)NCCN2CCC(NC(C(C=C)(C)O)=O)CC2)ccc2snnc2c1 c1(NC(=O)NC)ccc(C(=O)NC2CC2CNC(c2ccc[n+]([O-])c2)=O)c(Cl)c1 CC1=CCC(C(N2CCC(C)(NC(=O)CCc3cc(C)[nH]n3)C2)=O)CC1 C12(C(=O)NCCCN(C(c3cnc(C(N)=O)s3)=O)C3CC3)CCCN1CCC2 C(CCC(C(=O)NCC(F)Cl)NC(c1nonc1N)=O)OC Cc1[nH]nc(C(F)(F)F)c1C(=O)N(CCO)Cc1ccccc1N1CCCCC1 Cc1cc(NC(=O)CC2CCCN2C(c2ccccc2)=O)c(F)cc1Cl N1(C(C2CC(C)(C)OCC2)=O)CCC2(CC1)OCCC2NC(=O)CC1(CO)CC1 c1(C(=O)NCCC2(NC(C(CCOC)C)=O)CCC2)ccc(OC)cc1F CN1CCC(C(=O)NCC#CC(=O)NC2CCCC2C(N)=O)C1 c1(CC(=O)NC2C(NC(c3c(C)coc3)=O)COC2)ccccc1S(C)=O c1(NC(C2(C)N(Cc3c(OC)ncnc3OC)CC2)=O)nccc2scc(Br)c12 c1(C(=O)NCCC(C)N(C)C(c2cnc(S)[nH]2)=O)cc2c(nc1O)CCCC2=O C1(NC(c2cc(C)cc(O)n2)=O)CC2CC(C1)N(C(c1cc(N)c(Cl)cn1)=O)C2 C1(NC(C=COCC)=O)CCN(C(C2CCC(F)(F)C2)=O)C(C)C1 Cc1cc(Cl)ccc1OCC(=O)N(C1CCN(C(C2CC2C#N)=O)CC1)CCO C(C(=O)N1CCCC(C)(NC(=O)CCCC(N)=O)C1)(C(F)(F)F)OC(C)=O C1(CNC(CCC(C)SC)=O)CCCCCN1C(c1cnc(N(C)C)o1)=O N1(C(C2C(C#C)C2)=O)Cc2nccn2CC(NC(c2cnc(CC3CC3)s2)=O)C1 C1(N(C(C(C)N2CCCC2)=O)C)CCCN(C(c2cnc(C(F)F)s2)=O)C1 N1(C(c2cc(C)on2)=O)CCCCC(CNC(c2cnn(C3CC3)c2C)=O)CC1 c1(CC(C)NCC2CC(=O)N(Cc3ccccc3)C2)cc(Br)ccc1F C1(NC(CSC(C)(C)C)=O)CN(C(c2cncn2C2CC2)=O)CC12CC2 C1(CC(N2C(CC(=O)NCCn3ncc(C)c3)CC2)=O)CCOC1(C)C c1(CNC(c2cc(F)cc(F)c2)C(=O)OC)cc(F)cc(I)c1 c1(C(=O)NCC2CCCN(C(C(CC)n3cncn3)=O)C2)cc2ccccn2n1 CC1CCN(C(=O)C(C)(C)C(=O)N(C)C)CC1CNC(=O)C(C)(C)F C1(NC(C2C3CN(C(C(CC=C)(C)C)=O)C2C3)=O)CCC(=O)NC1(C)C CCCCCS(=O)(=O)CC(=O)N(C)CC1CCN(C(=O)C(C2CCCCC2)F)C1 c1(C(=O)NC(CC)CNC(=O)C=CS(F)(F)(F)(F)F)cnc2cc(O)ccc2c1 C(=O)(CC(C)(C)C)NC(C)C(=O)NCC#CCNC(=O)CCC1(C)CC1 N1(C(C(F)=C(C)C)=O)CC(C(=O)NCc2ccc(C#N)cn2)C(C)(C)C1 CC1CCCC(C(=O)N(CCCCCNC(=O)CC2(C3CC3)CC2)C)C1 C(=O)(C1CCc2snnc21)NC1(CNC(=O)Cn2ccnn2)CC2CCC1C2 c1(C(=O)NC(C)C(C)NC(c2ccc(N)c(Cl)n2)=O)cc2cccnc2cc1F Cc1c(Br)ccc(NC(C2(O)CCN(C(c3c(F)cc(Br)cc3Br)=O)C2)=O)c1F C(N=C(NC1CC1)N1CCC(O)C(C)C1)CC1=C(C)OCCS1 C1(C2CC2)(C(N(OC)Cc2ccc(C)o2)=O)CN(C(C23COCC2C3)=O)C1 c1(CNC(C2CCCN(c3cc(CO)ccn3)C2)C)nc(C)cc(C)n1 c1(OC)cc(C)cc(CNC2(c3cc(F)ccc3F)CC2)n1 C(=O)(C(C)CC(C)(C)C)NC12CN(C(c3cc(OC)c(C)cc3)=O)C(CC1)C2 C12(NC(C=CC=CC)=O)CCCCC1CN(C(C1CC3(CCC3)CO1)=O)C2 O=C1CCN(CC2CCCO2)C(=O)N1CC12CCC(CC1)OC2 N1(C(C(n2cc(Br)cn2)C)=O)CC2CC1C2NC(=O)Cc1ccns1 Cc1ccc(CNC(c2coc(CNC(c3ccccc3O)=O)n2)=O)nc1 c1(OC)ccc2c(c1)C(C(=O)N1CCN(C(c3ccnc(CO)c3)=O)CC1)CC2 c1(NC2(C)CC(NC(c3cnsn3)=O)C2)ccc([N+](=O)[O-])cc1CO Nc1cccc(C(=O)NCC2(CNC(=O)C(O)Cc3cnc[nH]3)CCCC2)n1 c1(C(N2C(CN(C(c3ccoc3Br)=O)CC)CCC2)=O)cc2n(n1)CCO2 C1(NC(C(=Cc2cccnc2)C)=O)CN(C(=O)Cc2nc(=N)[nH][nH]2)CCC1(C)C c1(C(N2CC(C)C(NC(=O)CC3CCC4CC34)C2)=O)c(Cl)nn(C)c1Cl C1(C(N2CCC(C(C)C)(C(=O)NC3CC(Cl)(Cl)C3)C2)=O)CC2CCC1CC2 C1(C(N(CC(=O)NC)CC)=O)CCCSC1.C(C(=O)OC(C)(C)C)CC(=O)N c1(C(N2CCN(c3nc(SC)nc(C)c3)CC2)=O)ccc(F)c(Br)c1F N1(C(c2cn(-c3scc(CC)n3)nc2)=O)CC2CC1CN(C(=O)CCC(N)=O)C2 CCN=c1[nH]cc(C(N2CC(O)(CCNC(C3CSCN3C(C)=O)=O)C2)=O)s1 C=C(C)C1OCCCC1C(=O)NCC(C(C)(C)C)NC(c1ccc(N)cc1Cl)=O C(CC#CC(C)(C)C)NC(C1(C#C)CN(C(C2CC2CCC)=O)C1)=O c1(C(=O)NCC2(NC(CC(C)n3cccc3)=O)CCOC2)nnn2c1CSCC2 C(=O)(CC1=CCCC1)NCC(C)C(=O)NCC1(C(N)=O)CC1 CC(C)(CCC(=O)NC1CCCCN(c2ncns2)C1)[N+](=O)[O-] c1(COC)cc(OC)ccc1N(C)CC1CCN(Cc2ccccc2)C1 CC1CC(c2cccnc2)N(C(=O)Cc2cccc(OC(F)(F)F)c2)C1 N1(C(C(C)OC)=O)CC(C)CN(C(=O)CCOc2cccc(Cl)c2)CC1C N1(C(C(=O)N(C)C)=O)CC2(CNC(c3cc(Cl)cc(F)c3N)=O)CCC1CC2 N1(C(c2cc(C3CC3)[nH]n2)=O)CCC(CCNC(C23CCC2C3)=O)CC1 N1(C(C(c2c(C)noc2C)CC)=O)CCOC(CNC(=O)CSCCC(C)C)C1 C1(C(=O)NCC2(CNC(=O)Cn3cnnc3O)CCC2)C2CC3C(C2)C13 N1(C(CCOCCN(C(CC2C(C)CCC2)=O)C)=O)CC(C2CCCC2)C1 C1(CC=C)(C(=O)NCCC(O)CO)CCCN1C(=O)CCOC(C)=O c1(C(N2CCC3(NC(=O)Cn4ncnn4)C(C2)C3)=O)cnc2ccccc2n1 c1(NCC(C)N(C(c2cccc(COC)c2)=O)C)ncnc2c1cnn2C(C)C C(CCC(C)C)(C(=O)NCCC(C)N(C(=O)COC(C)=O)C)NC(C)=O C1(C(N2CC(C)N(C(=O)COCCF)CC2)=O)CC2CCCCCC12 CC(C)CC(C)C(=O)NCCCN(C)C(C12CCC(C(F)F)(CC1)C2)=O C1(O)(CC(=O)Nc2cncc(Br)c2)CCN(C(c2cnc(Cl)s2)=O)C1 c1(CCC)ncc(NC(c2scnc2-c2cccnc2C(F)(F)F)=O)cn1 CCCC(C(=O)N(CCNC(c1ccnc(C)n1)=O)Cc1ccccc1)OC O=C(C1SCCc2ccccc21)NCC1CCN1C(=O)CC=Cc1ccccc1 CCCC(C)CC(=O)NCC(CC1CC1)C(=O)N(CC(F)F)CC(C)O c1(CN(C(C)=O)Cc2cccc(Cn3cccn3)c2)nc(C)c(CC2CCCC2)s1 C1(CC)CCCN(CC(=O)Nc2cccc(C(=O)N(C)Cc3ccccc3)c2)C1 C1(CCOC)CN(C(=O)C=CC(C)C)CCN1C(=O)CCCN=[N+]=[N-] C(CCCC(F)(F)F)NC(C(c1cn(C)nc1)NC(c1cc(CO)on1)=O)=O CC1=C(C)CC(C(N2CCC(OCCNC(=O)Cc3cc(C)sc3C)C2)=O)CC1 C1(C(=O)NCCC2CC(NC(=O)Cc3cc[nH]c3)C2)Cc2c[nH]cc2S1(=O)=O CCCCCC(O)C(=O)NC12CCCN(C(c3cnc(=NCC)[nH]c3)=O)CC1C2 c1(CNC(C2N(C(c3c(C)c(I)ccc3)=O)CCOC2)=O)cc(Cl)c(F)c(Cl)c1 C1(CNC(c2n(CC)nnc2)=O)CC(O)CN1C(c1ocnc1C1CC1)=O c1(C(C)NC2CCC(OCC(N3CCCC3)=O)C2)cc(Cl)sc1Cl c1(C(=O)NCC2CCN(C(C=CC)=O)CC2)cc(F)c(Br)cc1[N+](=O)[O-] c1(C(N2CC(OC)(CNC(c3n[nH]cc3Cl)=O)C2)=O)ccc(-n2ccnc2)cn1 C1(C#N)(C(=O)NCC(CC)NC(=O)C(C)COC)CCS(=O)(=O)CC1 Cc1cnn2c1CN(C(=O)C(=O)NCCOC1CCCCC1)CC2 C(=O)(C1COCc2ccccc21)NC(C1CCCC1)CNC(=O)Cc1nc[nH]n1 C(N=c1[nH]c(=NC(C)C2CCC2)[nH]c2cc[nH]c12)c1cc(OC)c([N+](=O)[O-])cc1 c1(C(=O)OC)cccnc1NC1CCCN1C(=O)C(c1ccc(Cl)cc1)OC N1(C(C(C)=C2CC2)=O)CCC2CC(CNC(C3CC(C)(F)C3)=O)CCC2C1 c1(CC)cc(Cl)ccc1C(=O)NC1C=CCN(C(=O)CCNS(C)(=O)=O)C1 c1(CC(=O)NCCC(C)N(C(=O)CC(C2CCC2)C2CCC2)C)nn(C)cc1Cl C1(C(N(C(C#C)C)C)=O)CC2(CC2)C12CCC2 CCCCCC(C)CC(=O)NC1CCN(C(=O)CC2CN(C(C)=O)C2)CC(O)C1 N1(C(C2(C(=O)NC)CC2)=O)C2CCC1CN(C(=O)C(c1ccc(Cl)cc1)=O)C2 C1(C(=O)NC2CC(OC(C)C)C2)N(C(C2CCCCC(=O)N2)=O)CCCC1(C)C C(=O)(C1=C(C)OCCC1)N1C(C(N(CC(CC=C)(F)F)C)=O)C2CCC1C2 c1(C(=O)NCC(C)CN(C)C(C2CS(=O)(=O)CCO2)=O)cnn2cccnc12 C1(CC(=O)NC2(C(=O)NCCNc3cc(Cl)c[nH]3)CCC2)COC(C(F)F)C1 c1(CC(=O)NCCN(C(CC(=C=C)C)=O)C2CC2)ccc(F)cc1C N1(C(CCC(C)NC(C23CC(C#N)(C2)C3)=O)=O)CC2(COC(=O)N2C)C1 c1(C(=O)NCCC(C)NC(C2CC(C#N)C2)=O)cc(C2(C)CC2)n[nH]1 C1(NC(c2c(C)cc(C)s2)=O)CC(C)CN(C(=O)CC2CCCC(C)(C)O2)C1 c1(C(=O)NCCNC(C(CCC)O)=O)cnc(C)c(Cl)c1Br C1(C(=O)NCC(C)(C)N(C)C)CCN(C(c2cc3ccccc3[nH]2)=O)C12CCC2 c1(C(N2CCCC(CCNC(C3(C)CCOC3)=O)C2)=O)ccc(P(C)(C)=O)o1 C1(c2ccc(OC)cc2)CCc2nc(O)c(C(=O)OCC(Br)Br)cc2C1 N1(C(C(C(C)CC)NC(C(C2CCC2)OCC)=O)=O)CCC(C2(C)CC2)C1 c1(C(=O)NC2CCC(CNC(C3C(C)(C)C3(F)F)=O)C2)c(N)cccc1F N1(C(CC(C)O)=O)CCCCC1CCC(C)(C)NC(=O)CCc1cccc(F)c1 Cc1cc(C(=O)NC2CCC(NC(C3(C)CC3Br)=O)CC2)cc(C)c1Cl c1(CC)cccc(C(N2CC=CC2CNC(c2csc(-c3ncc[nH]3)n2)=O)=O)n1 N1(C(CN(C)C)=O)CC(F)CC1CNC(C1CC1c1ccco1)=O C(=O)(C1=C(CC)OCCC1)N1CC(NC(c2c(Cl)ccc(C#C)c2)=O)C(C)C1 CN1C(=O)CC(C(=O)Nc2nnc(CC(F)(F)F)s2)NC1=O c1(C(=O)NCCN(CC(C)O)C(c2cnc(C(C)C)[nH]2)=O)cnc(Cl)c(F)c1N c1(OC)cccc(CC(=O)OC(C)(CC(=O)O)c2cccc(F)c2)c1F C=C1C(C(=O)NOCC(=O)NCC(C)(C)OCC)C1C(=O)O c1(C(=O)NC(CNC(CC2CC(SC)C2)=O)CO)ccnn1C1CC1 N1(C(C(CC)F)=O)CCC2CC1CN(C(c1ccc3[nH]ccc3c1)=O)C2 N1(C(c2cc(C#N)[nH]c2)=O)CCC2(C1)CN(C(=O)C(F)=C1CCCC1)CCO2 c1(-c2c(OC)cccc2F)ccc2[nH]c(C(=O)Nc3ccnn3C(C)C)nc2c1 N1(C(C(CC=C)C)=O)C2CC1CN(C(=O)Cc1ccccc1CC(N)=O)C2 CC(C(=O)NOCCCOC(c1ccc(Cl)cc1)=O)C(C)SC(C)(C)C c1(OC)ccc(N(C(=O)Cc2ccc(F)cc2)C)cc1 C1(C(C)C)CN(C(C23CC(C)(CO2)C3)=O)CCN1C(=O)CCc1ccsc1Cl N1(C(c2n(CC)nnc2)=O)CC(C2CCCN(C(C3C4CCCOC34)=O)C2)C1 CC(C(=O)NCc1cn[nH]c1)(C1CCC1)NC(=O)CCc1ccccn1 N1(C(C(C)N(C(=O)CC23CCCC2C3)C)=O)CCSC2(CCC2)C1 C1(N(C)C(C2(CO)CCCC2)=O)CCCCC1NC(=O)C(c1ccccc1)F C(=O)(CCC(=O)OC)NCCN(C(=O)C(C)N1CCC1)CC(=C)C Cc1cc(F)c(N)cc1C(=O)NCCC(O)CNC(=O)C1=CCCOC1 C1(C)(C(=O)NC2C(NC(c3c(C(C)C)ncs3)=O)CC2)CCCCNC1=O c1(C(=O)NC2CC(F)(CNC(=O)CCC3CCCC3)C2)ncccc1C(F)(F)F CN1CCN(C(c2cc(N)cc(O)n2)=O)C(CNC(=O)CC2CCCCC2O)C1 C(CCC(C)(C)C(=O)N1CC(C)(C)C1C(=O)OC)NC(C(CC=C)OC)=O C1(CCNC(C(CCOC)(C)C)=O)CN(c2nnc(C(N)=O)s2)CCS1(=O)=O C#Cc1cccc(C(=O)NCC2(C)CC2C(=O)N(C)Cc2cc(C)n(C)n2)c1 CCCCC(CC(=O)N1CCCCC1C1(O)CC1)NC(c1ccc(C#N)[nH]1)=O c1(CCC(=O)NC23CN(C(C4CC=C(C)CC4)=O)C(C2)C3)cc(F)ccc1F C1(C(N(C(c2cccnc2)C)C)=O)CN(C(c2ccsc2)=O)CC1(F)F c1(COc2ccccc2)nc(-c2cc(C3CCOC3)[nH]n2)n(-c2nc[nH]n2)n1 C1(C(=O)NC2(C)CCCCC2)CC2CCCCC2N1c1ncc(C(F)(F)F)cn1 CC1(C)CCC(C(=O)NCC(C2CCCC2)NC(=O)C(C)(C)c2cc[nH]n2)C1 C1(NC(c2[nH]ccc2CNC(C2C3CCCC(=O)C23)=O)=O)CCCN2CCCC12 Cn1cc(C(N2CCC(NC(=O)CC3CCSC3)C(F)C2)=O)ccc1=O N1(CC(N2CCC(O)(CNC(C(C)C3(O)CCC3)=O)C2)=O)CCP(C)(=O)CC1 c1(C(C(=O)NCC2C(CNC(CCC#N)=O)C2)O)ccccc1Br C1(N(CC(C)C)CC#C)(CNCC(=O)Nc2cnoc2C)CCCCC1 S(=O)(=O)(c1cc(C(=O)N(CC(C)C(C)(C)C)C)co1)NC C1(C#N)(C(N2C(CN(C)C(c3scnc3C(C)(C)C)=O)CC2)=O)CCCC1 C(CC(CC)C(=O)NCC(C)(CC)C(=O)NCCCCCCO)=CC N1(C(C2C(C)C2)=O)CCN(C2CN(C(=O)COCC3(F)CC3)C2)CC1 N1(C(C2(C)CC(C)C2)=O)CC2CCCC2(NC(c2cc(C)c(C)[nH]2)=O)C1 c1(C(=O)NC2C=CCN(C(C3N(CC)CCOC3)=O)C2)cc(O)ncc1Br Cc1ncc(Cl)cc1C(=O)N(C)C(=O)NCC(C(F)(F)F)n1cncn1 c1(OC(C)C(=O)NCCN(C2CCCC2)C(c2cc(F)c[nH]2)=O)ccccc1F c1(C(=O)NC2CCCCC2NC(C2C=CCC2)=O)cnc2ccccn2c1=O c1(COCC)c(C)nc(O)nc1C.C12(C(=O)OC(C)(C)C)CCCN1C(=O)NC2 c1(C(=O)NC2CC(O)CN(C(c3scnc3C3CC3)=O)C2)cc2cnccc2[nH]1 CCC(CO)C(=O)NC1CN(C(C2(c3ccc(C)nc3)CC2)=O)CC1C N1(C(C(C)(C)c2cccnc2)=O)CCOCC(CNC(=O)Cc2cnc[nH]2)C1 C1(OC)CCCC(C(=O)NCCC2(Nc3cnccc3Cl)CCC2)C1 C1(C)(CNC(c2c(OC)ccnc2O)=O)CN(C(=O)CCCC(N)=O)C(C)(C)C1 c1(C(=O)NC2(C)CCN(C(=O)C=C3CCCCC3)CC2)ccc2ncccc2n1 C(=O)(CCCC(C)(F)F)NC1(CC=C)CCN(C(=O)C(C(C)(C)C)NC(C)(C)C)C1 CC1(C)OCC(c2cn(CC3CCCC3NC(C3(n4cnnn4)CC3)=O)nn2)O1 C12(NC(COCCCCCC)=O)CCN(C(=O)Cc3csc(C(C)C)n3)CC1C2 C1(NC(C2C(C)(C(C)C)C2)=O)COCCN(C(C2(C#N)CC3CC3C2)=O)C1 C1(NC(C2(NC(C3CCCO3)=O)CC(CO)C2)=O)CCC2(CCCC2)C1 C(=O)(C1CCc2c[nH]nc21)NC1C=CCC(C(N(C2CCCCC2)CC)=O)C1 N1(Cc2nc(C)c(C)s2)CCC12CCCC(C)(C)C2 c1(OC)nc(C(N2CCCC(OCc3ncc(C)[nH]3)C2)=O)cc2ccccc12 c1(N2C(C)CCC(C)(C)C2)cc2ccncc2cn1 c1(CC)ccc(C)c(C(=O)NCC(C2CCC2)NC(=O)CCC2CCC(=O)C2)c1 c1(C(=O)NC(CN(C(c2c(C(C)C)onc2C)=O)C)C)cccc(O)c1F C(=O)(CCC(=O)N1CC(CNC(=O)C=CCOc2ccccc2)CC1C)NC c1(N(CC(C)C)C)nnc(C2CC2)n1NCC1CCSC1(C)C N1(C(C(C)C2CC2)=O)CC(C(=O)NCc2ccccc2O)CCC1(C)C N1(C(=O)Cc2csnn2)CCC2(CCCN2C(c2cc(C3CCC3)no2)=O)C1 C(C)(C)(CCC(=O)NCCc1noc(C)n1)NC(Cn1nnc(C)n1)=O N1(C(c2c(SC)ccs2)=O)CCC(NC(=O)C(C)Cn2ccc(C)n2)C12CC2 C1(NC(C2NC3CC2C3)=O)CCC(OCCF)CC1 Cc1nc2cc(C(=O)NCCC3CC(NC(=O)CCc4cnc[nH]4)C3)ccc2s1 N#Cc1cccc(N(C(C2CCC(C#N)CC2)C(=O)NC2CCC(F)(F)CC2)C)c1 c1(C(N2CCC(O)(C(C)NC(=O)C=CC3CCCC3)C2)=O)c(Cl)ccc(Cl)c1O N1(C(C(=O)NC(C)C)=O)CC(NC(C2CCC(F)CC2)=O)C(C)C1 C1(N(c2ccc3cccnn23)C(C)(C)C)COC2CN(C(=O)C(O)P(C)(C)=O)CC12 C=CCCN=C(NCC1CC=CCO1)NCC(C(C)C)c1cccnc1 c1(-c2n(C(COC)C)nc(-c3cccc(OC)c3)n2)ccc(Br)c(Cl)c1 CCCC(CC)C(=O)N1CCOCC1(C)c1cn(Cc2cc(C)nc(C)c2)nn1 C(C1=CCN(C(=O)CC2CC23CC3)CC1)NC(=O)Cc1cc(Cl)sc1Cl c1(CC(=O)NC2(COC)CN(C(C3N(CC)CCC3)=O)C2)nn(C)cc1Cl Cc1cc(C(=O)NCC2CC(C)N(C(c3ccco3)=O)C2)cc(C)c1 Cc1cc(C(N2CCC(C)C(CNC(=O)C(C)(C)CO)C2)=O)c(Cl)cc1F C(C(C)(C)C(=O)NCCC1CCC(C)(C)O1)N(C(=O)CCC1CCCOC1)C N1(C(N(C2CCCCC2O)C)=O)CCCCCC1c1ncon1 C(CC(C(=O)N=c1ccn(CC2CC2)[nH]1)N(C)C)NC(C1=C(C)CCC1)=O C12(NC(C(CCC)C)=O)CC(C)(C1)OC21CN(C(C2CNC(=O)CC2C)=O)C1 C1(COC)(CNC(C23CCCC2(C(N)=O)C3)=O)CCN(C(=O)CC(C)F)C1 c1(C(C(=O)NCCC2CCC(NC(CC3(C#N)CC3)=O)C2)=O)ccc(Cl)cc1 C1(CC)CCCCC1OCC(N1CCC(NC(=O)C=Cc2sccc2C)C1)=O Cc1cc(Br)ccc1C(N1CC(CNC(C2CCC(C(N)=O)C2)=O)C(C)C1)=O c1(C(N2CCC(C(C)NC(c3c(C)nncc3)=O)C2)=O)ccc2c(ccn2C)c1 CC1=NOC(=O)C1CCC(=O)NC(C)CNC(c1oc(C2CCC2)nc1C)=O CC1Cc2cc(C(=O)NC3CCCN(c4nc(Cl)ncc4F)C3)ccc2O1 c1(NCC2(O)CCN(C(c3ccc(C(C)O)cc3)=O)C2)cccc2nccn12 N1(CC(=C)Cl)CCC(C2CCN(C(c3csc(O)n3)=O)CC2)C1 C1(CCNC(CN(CC(C)(C)C)C)=O)CC(NC(=O)CC2(C#N)CC2)C1 c1(C2(C(N3C(CNC(c4sccc4Br)=O)CCC3)=O)CCCC2)ccc(Br)cc1 C(=O)(C(C)(C)C(=O)NC1CC(CC(=O)NCC2CS(=O)(=O)C2)C1)OC N1(C(C2(C(CC)=O)CC2)=O)CCC(C(=O)NCC2CCC(C)C2)=C(F)C1 N1(C(C(C)OC(C)C)=O)CCOC2(CCN(C(=O)CCn3ccnc3)C2)C1 N1(C(C2(C)CC=CC2)=O)CCCC(O)(CCNC(c2occ3c2CCC3)=O)C1 CN=c1[nH]c(=NCc2ccc(SCCCO)cc2)[nH]c(=NC2CCSC(C)C2)[nH]1 C1(C(=O)O)CCN(C)C1.n1(C2(C(=O)NC(=O)CC3(C4CC4)CC3)CC2)cc(Cl)cn1 N1(C(c2c(CC)ccs2)=O)CCCC(CCNC(c2cccc(OC)n2)=O)C1 C1(C)(C(=O)NC(COC(C)=O)CO)CN(C(=O)C(C)C#N)C1 C1(NC(C2CC3(C2)CC3F)=O)CCN(Cc2cn(CC3CC4CC4C3)nn2)CC1 N1(C(C(CC)(C)O)=O)C2CCC1CC(C(=O)NCc1csc(C)n1)C2 CC(Cc1ccco1)N=c1nc(N2CC(F)C(F)C2)c2[nH]ccc2[nH]1 CCCC(C)CC(=O)N1CC2C(CNC(c3c[nH]nc3-c3cccs3)=O)C2C1 C1(NC(C2NC(=O)OC2)=O)CCCC(NC(C2COCCOC2)=O)C1 c1(C(=O)OC)[nH]c2ccccc2c1C(N1CC2CC(N3CC4CC4C3)C1C2)=O N(C1CCc2ccc(Cl)cc21)C(=O)CC1CCCCC1(F)F c1(C(N(CCCCNC(c2nc(CC)oc2C)=O)C)=O)cc2n(c1)CCCC2 c1(C(=O)NCCN(C(=O)CC2CCCC2O)CCC)nocc1Br C1(=O)C(C)CN(C)C(=O)CN2CC(C)(C2)N1C(C)C(C)C.COC N1(C(C=COC(N2CCC(C(=O)NC)C2)=O)=O)CCC(CC(C)OCC)CC1 N1(C(C=Cc2n(C)ccc2)=O)CCC2C(C1)CN2C(=O)C(C1CCOCC1)F C=CC(C)(C)C(=O)NC1CCCC1NC(c1ccccc1SCc1cscn1)=O C(c1cc(Cl)cc(Cl)c1)=CC(=O)NC(CC(=O)OC)Cc1ccc(C)cc1 C1(CCC(=O)NC2(C3CC3)CCC2)CCCN(C(C23CCCC2C3)=O)C1 CC(C)CC(C(=O)NCC1C(C)CCN1C(c1cccc(=O)n1O)=O)N(C)C N1(C(CCOC(C)=O)=O)CCC2CC12C(=O)NCC(CO)C1CC1 c1(OC)cn(CC(N2CCOCC2CNC(=O)C(C)P(C)(C)=O)=O)c(C)cc1=O Cc1cc(N2CC(O)CC2C(=O)NCCOc2ccccc2Br)ncn1 C(CNC(=O)CN1CCC(C)CC1)(C(=O)NOC(CC)CC)OC CC(O)(CC(=O)NCC1CCCC1NC(C1(CC2CC2)CC1)=O)C(F)(F)F C1(CNC(c2cnn[nH]2)=O)CCC2CN(C(=O)Cn3cnccc3=O)CCC2C1 N1(C(c2c(CC)ncs2)=O)CCOCC1CC(=O)NCCCc1nc(C)no1 Cc1nc(C(=O)O)ccc1C(=O)NC(c1cn(Cc2ncccn2)nn1)C CCC(C)(C)C(=O)C(=O)N1CCN(C(c2cn3c(n2)CCCC3)=O)CC12CC2 C=C(C)CC(C(=O)N1CCCC1(C)CNC(c1nccc(C)n1)=O)OC CC(C)(C)CC(C)(C)C(=O)NC(CNC(c1n[nH]c2c1CC1CC21)=O)C1CCC1 N1(C(=O)OC(C)(C)C)CCCC(C)(NC(N2CC(CCO)(CO)C2)=O)C1 C1(C(N2C(COC)CCCC2)=O)N(C(=O)C=Cc2ccc(C)o2)CC12CCCC2 C1(CNC(CNC(C2(CC)CCC2)=O)=O)CCCOCC1.C1C(=O)NCCO1 Cc1cc(C(N2CC3CC3(CNC(C3(C)CC4CC4C3)=O)C2)=O)nc(C)c1 C(=O)(C#CC1CCCO1)N(C)Cc1ccco1.C12CCCCN1C(=O)CNC2=O c1(C(=O)NCC(CCNC(C(C=C)(C)C)=O)=C)cccc2ncnn12 N#Cc1cc(F)ccc1C(N1CCC2(CC(NC(C3CCCS3(=O)=O)=O)C2)C1)=O CC(C)(N=[N+]=[N-])C(=O)N1CCCCC(CCC(=O)NCc2cc(O)cc(F)c2)C1 c1(C(=O)OCC(=O)NCC2CCC3CC23)nsc2cc(Br)ccc12 N(C(=NCCC1(O)CCC1)NCCN1CCCC1)CC(c1ccc(C)cn1)O N1(C(C2(C(C)C)CC2)=O)CCC(C)(C(=O)NCc2cnccc2Cl)C1 N1(C(CCCC(C)O)=O)CCCC(C2CCN(C(c3nn(C)cc3Cl)=O)CC2)C1 C1(NC(CCC(N)=O)=O)CN(C(=O)COCC2CCCC2)CC2(CC2)C1 O=C1CCC(CC(=O)NCCc2n[nH]cc2C(=O)NC2(c3nn[nH]n3)CC2)CC1 C1(CC)CN(C(=O)CC(C)(C)N(C)C)CCN1C(=O)CC1(C)CCCC1 C1(CCNC(c2nccc(C)c2)=O)CCN(C(C2(C)CNC(=O)N2)=O)CC1(F)F C=CC(F)(F)C(=O)NC(C)CN(C(=O)C(C)Cc1cnco1)CC C(=O)(C(C(=O)OCC)NC(=O)NC1(CC(=O)OC)CCC1)OCC CC(C)(CNC(=O)Cc1n[nH]c(=N)s1)CCNC(c1cncc(Br)c1)=O C=CCCN=C(NCC1COC(C)(C)C1)NCC1CCC2(CCCC2)O1 c1(C(=O)NC(C(CO)NC(c2c(OC)nsc2)=O)C)cc2sccc2cn1 C#Cc1cn(C)nc1C(=O)NCC1(CN(C(=O)CNC(=O)C2CC2)C)CC1 Cc1ccccc1C=CC(=O)NC1CCC(CNC(=O)C(C)CC2CC2)CC1 C1(C(N(CCC(C)C)CCC#N)=O)Cc2ccccc2CN1C(C1(C)CC1)=O C(=O)(CC(F)(F)CC(=O)NC1COCC1NC(C1COCCN1C)=O)OC CC1CN(c2ccc(CNC(c3n[nH]cc3F)=O)cn2)CCO1 c1(NC(=O)CCC(=O)C2CC2c2ccc(Cl)cc2)ncccc1C=CC(F)(F)F N1(C(c2cncc(OCC)c2)=O)CCN(C(c2c(CO)n[nH]c2C)=O)CC1C N1(CCNC(CCCOC)=O)CCCN(C(=O)C(c2ccccc2)N(C)C)CC1 CCCCCS(=O)(=O)CC(=O)NCCCC(C)(C)NC(=O)CC(CC)OC N1(C(C=CC)=O)CCC(c2ccccc2)(NC(c2cc(C)co2)=O)C1 C1(NC(COc2cn(C)nc2)=O)CCN(C(c2ccoc2)=O)CC1 c1(C(N2CC(C)(NC(c3ccc(N(C)C)cc3)=O)C2)=O)cc2n(n1)CCCC2=O C1(C(=O)NCC(Cc2ccccc2)NC(C(F)OC)=O)CCCCC1O C1(CN(C(c2ccc(SC)s2)=O)C)COCCN1C(C1CCCN1C1CC1)=O CC1CN(C(C2OCC2(C)C)=O)CC1CNC(c1ccnc(CN(C)C)c1)=O C1(CCC(C)(C)NC(C(CC)=CC)=O)CCN(C(c2cc(F)n(C)n2)=O)CC1 c1(C(C(=O)N(C)CC2CCCCN2C(C23CC(C2)C3)=O)O)cc(Cl)cc(Cl)c1 Cc1nocc1C(=O)NC1CC(O)(CNC(c2cccs2)=O)C1 C1(O)(CNCc2nccc(OC(C)C)c2N)CCCC12CCOCC2 N1(C(CC(c2cccc(F)c2)C)=O)CCN(C(c2cnc(Cl)s2)=O)CC(O)C1 C(CN=c1[nH]c(=NCCC(C(C)(C)C)OC)[nH]c2cc[nH]c12)N(C)CC c1(C(=O)NC2(CNC(C(C)C3CCCO3)=O)CCCCC2)cncc(O)c1Cl C1(c2c(C)ccnc2)CCN(C(=NCC(C)C)NCC2(C(N)=O)CCCC2)C1 C1(C(=O)NCC(C)(C)CSC)(COC)CN(C(=O)CCC2CC2(F)F)C1 N1(C(CSCC(N)=O)=O)CCC(NC(=O)CC2(Sc3ccccc3)CC2)C(F)C1 c1(SCC#C)cccc(C(N2CC(NC(C3(OC)CC3)=O)C(C)C2)=O)c1 C#CCCCCCCC(=O)NC1CCC(CCC(N2CCCC(C(N)=O)CC2)=O)C1 C#CCC(C)C(=O)NCC(F)CNC(=O)CCc1ccc(C(F)F)cc1 c1(C(N2CC(NC(c3cc(CC)[nH]n3)=O)C(F)CC2)=O)cnc2snnc2c1 C1(CCCNC(C(n2cc(C(=O)O)cn2)C)=O)(CN)CCCC1 C(CCCCC(=O)N1CCSC2CCC12)NC(c1cc(CCC)[nH]n1)=O n1(CC(=O)NC2CC(NC(CC)=O)C23CCC3)cc(C)c(O)nc1=O CCCCCC(CC)C(=O)NC1CC(CCNC(c2ncccc2F)=O)C1 c1(-c2cc(OC)c(OC)nc2)ccc2sc(C(=O)Nc3c(C)noc3C)cc2c1 N1(C(c2c(NC)cnnc2)=O)CCN(C(=O)C(=Cc2ccc(F)cc2)C)C2CC12 Cc1[nH]nc(C(N2CCC(O)(CN(C)C(c3cncnc3)=O)C2)=O)c1Cl C1(C(=O)NCC2(OCCNC(C3CC3Cl)=O)CCOCC2)CC2(C1)CC(F)(F)C2 c1(CCC(=O)N2CC(CNC(=O)C(O)CC3CC3)C2)ccc(O)cc1 c1(C(=O)NC2CC(NC(=O)C(F)F)C2)ccc(-c2ccc(Cl)cc2)cc1 c1(C(N2CCC(N(C(=O)C3CC3)Cc3ccccc3)C2)=O)nccn1C1CC1 CCCC(C(=O)N1CC(NC(c2cc(S(N)(=O)=O)cs2)=O)C2(CC2)C1)C(C)C C(=O)(CC(C)(C)C(C)(F)F)N1C(C)CC(NC(c2ccc3cncn3c2)=O)C1 N1(C(c2c(C)cns2)=O)Cc2ccccc2CC1CNC(C1CCCOC1)=O c1(N2CC3(C(NC(c4c(C#N)cn[nH]4)=O)CCS3)C2)ccc([N+](=O)[O-])cc1[N+](=O)[O-] CCCC(O)CC(=O)NCc1ccccc1CNC(C1(F)CC=CC1)=O C#CCC(C(=O)N1CC(C2CCCO2)C1)NC(C1CC2CC2C1)=O C#Cc1cnn(CC(=O)NC2CCCCC2NC(C2CCCN2C(C)=O)=O)c1 C1(O)(CNC(c2cc(Br)c[nH]2)=O)CCCN(C(c2ccc(Cl)cn2)=O)C1 C1(CC(=O)NC(C2CC(F)(F)C2)C)C2CCC(C2)N1C(=O)CN1CC2CC2C1 c1(OC)ccc(C)c(C(=O)NCCC2CN(C(C3(C4CCC4)CC3)=O)CC2C)c1 N1(C(c2c(OC)c(C)sc2)=O)CCN(C(=O)Cc2ccc(C)c(O)c2)C(C)C1 C(=O)(CCN(OC)C(=O)c1ccsc1C)N1CC(C#C)C1 n1(CCOC)ccc(C(=O)NCC2CC(CNC(C3C(C)C3C)=O)C2)n1 C1(NC(C2CCC3CC3C2)=O)CCC2CC1CN2C(=O)CC1CCC(=O)N1 N1(C(C2(NC(=O)OC(C)(C)C)C(C)C2)=O)CCS(=O)C(C)(C)CC1 c1(C(C)NC(C=CC(C)NC(=O)C(Cl)=CCl)=O)cccnc1O N1(C(c2cc(C(C)=O)sc2)=O)CCC2CN(C(c3cc4n(n3)CCC4)=O)CC2C1 C1(CCN(C)CC2CCOC2)CCN(C(=O)Cc2ccccc2Br)CC1 c1(C(N2CCC(c3nnc(C)s3)CC2)C(=O)NCCOC)nc(Br)ccc1F C1(C(=O)NC(COC(c2cc(C)sn2)=O)=O)CC2CC(=O)C1O2 CC12CC(CC(N3CCCC(CCNC(=O)C4=CSCS4)C3)=O)(CO1)C2 Cc1ccc([N+](=O)[O-])cc1C(N1CCCC(C)(NC(C2CCCCC2)=O)C1)=O C(c1ccc(O)cc1)=CC(=O)N(C(C)CNC(C1CN(S(=O)(=O)CC)C1)=O)CC c1(C(=O)NCC(C(C)C)NC(C(CCC)C#N)=O)nc2ncc(C)cn2n1 CCC(CC1CCCC1)C(=O)NC1CC(C)(NC(c2ccnn2C2CC2)=O)C1 N(C1CCCc2[nH]ccc21)C(c1c(C)cc(Cl)c(Cl)c1)=O C1(CNC(c2cnc(CC)[nH]2)=O)C2CCC(C2)N1C(c1ccc(C#N)o1)=O N1(Cc2onc(C)n2)CCOCC(C(=O)N(C)Cc2noc(C(F)(F)F)n2)C1 c1(C(N2CC3C(NC(=O)Cc4ccsn4)(C3)C2)=O)ccc2cccnc2c1F CC1CN(C(=O)Nc2cnn(-c3cccc(F)c3)c2)CC2(CCOCC2)O1 c1(N2CCC(CC)(CO)CC2)ncc(S(=O)(=O)N(C)CC2CCOCC2)cc1Cl c1(C(=O)NCC2C=CC(NC(C(CCCC)O)=O)C2)ccc2c(c1)CCN2C=O C(=O)(C1CCCc2c(O)cccc21)N1CCCN(C(C2(C)CC2)=O)CC1CO c1(CNC2C(C(=O)Nc3c(OC)ccc(C(N)=O)c3)C2)cccc([N+](=O)[O-])c1 N1(C(CC2C(C)(C)C(O)C2)=O)CC2CC(NC(c3cc(Cl)c[nH]3)=O)CC1C2 C1(NC(c2cc(C)nn2C)=O)CCN(C(C2CCC(=O)C(C)C2)=O)CC12CCC2 c1(C(=O)NC2CC2)ccncn1.C1(C(N2CCCC2)(C)C)CCCN1C(=O)C=CCF C1(=CC(=O)NCC2(C)N(C(CCSCC(C)C)=O)CCC2)CN2CCC1CC2 Cc1cc(CC(=O)NC(CNC(C2CC3OC2C2CC32)=O)C(C)C)cc(O)n1 CCC(CC(C)C)C(=O)NC12CC1CN(C(=O)C=Cc1nc(C)c(C)[nH]1)C2 C(=O)(CCCC(=O)NC1CN(C(=O)CCn2cccn2)C(C)(CC)C1)NCC N1(C(=O)Cc2ccc(Br)cn2)CC2CN(Cc3ccccc3I)CC2C1 c1(NC(N2CC(F)(c3ccccc3)C2)=O)ccc(-c2cncnc2)cc1F n1(CC#C)cnnc1C(=O)NC1(CCC(=O)N(C)Cc2cncs2)CCCC1 C1(CNC(COC(C)C)=O)(CNC(=O)CCc2cn(C)nn2)CC12CCC2 C1(CCNC(c2cocc2C)=O)(NC(C(C2CC2)SC)=O)CCOCC1 C(=O)(C(C(C)C1CC1)N1CCC(CSC)C1)NCCSC C1(C(N(CCCNC(c2c(C)cc(=N)[nH]c2)=O)C)=O)CCc2ccnn2C1 C12(CNC(=O)CSCCC3CCCCO3)CC1CN(C(C13CC(F)(C1)C3)=O)C2 CS(=O)CCC(=O)NC1C=CCN(C(c2cc(COC(C)(C)C)on2)=O)C1 C1(C(=O)NC(CNC(c2c(C)cccn2)=O)(C)CO)CCS(=O)(=O)C1(C)C C1(N(C2CCCCO2)C(c2cc(COC)[nH]n2)=O)C2CCC1CNC2 C1(NC(c2c(C)ccs2)=O)CN(C(c2c[nH]ccc2=N)=O)CC2(CC2)C1 C=Cc1ccc(C(=O)NCCOC2CN(C(c3cnn4cc[nH]c34)=O)C2)cc1 N1(C(CCC2C(C)C2)=O)CCN(C(=O)C(C)(C)C2CC2)CC1 c1(CC)oc(C(=O)NC(C2CC2C(=O)NOCc2ccccn2)C)cc1C C(=O)(C1=CCCCCC1)NCC1N(C(C(C)=CC2CC2)=O)CC(F)(F)C1 N1(CC)C2CCC1CN(C(=O)CNC(C)=O)C2.c12nn(C)c(c1Br)NC2=O N1(C(COC2CC(N(C)C)C2)=O)CC2CC(C1)N2C(=O)C(C)(Cl)Cl C1(CC(N2CCC2CCc2[nH]nnc2C)=O)CCN(CC)C1 c1(CNC(c2nnnn2CCN2CCOCC2)C2CC(=C)C2)cnc(C(C)C)o1 C(=O)(C1CCc2ccccc21)N(C(C)C(N1CCN2CCCCC2C1)=O)CC c1(CN(C(C2CCN(C(C3(CC)CCCCO3)=O)C2)CC)C)ccccc1Cl c1(CN2CC(NC(c3ccc(Cl)o3)=O)C(O)C2)ccc(F)cc1[N+](=O)[O-] c1(CC)nc(C)c(C(=O)NC2COCCC2NC(=O)CC(CC)SC)s1 Cc1cncc(F)c1C(=O)NC1CC(CNC(=O)CN2CCCC(N(C)C)C2)C1 c1(C(C)=O)c(C)[nH]c(C(=O)NC(C)CNC(=O)CCSc2cccc(C)c2)c1C c1(C(=O)NCCC2CN(C(=O)CCN3CCOCC3=O)C2)cc(F)c(F)cc1O N1(S(CC)(=O)=O)CCCC(C(=O)Nc2ccccc2CNC2CCOC2)C1 N1(C(Cc2ccc(C)s2)=O)CC2(COC(CNC(C3(C)CCC3)=O)C2)C1 Cc1cc(C(=O)N(CC(C)NC(c2cn(CCF)nn2)=O)C)c(C)c(C)c1 c1(C(N(CC(CN(C(C(C)=C(C)C)=O)C)O)C)=O)csc(C(F)(F)F)n1 C(CNC(=O)CSCCC(C)C)(CC(C)C)NC(c1cnc(OC)s1)=O CC(CCNC(c1ccc(-c2cccnc2)cn1)=O)CCNC(=O)C1=CCOC1 c1(CS(N2CCC(C(=O)NCc3cc(Br)no3)C2)(=O)=O)ccc(Cl)c(Cl)c1 CC1(C)NC(=O)CC1C(N1CCCC(O)(CCNC(C2(S(C)(=O)=O)CC2)=O)C1)=O C1(C(=O)NC2CC(OCC(=O)NC3C(C=C)COC3)C2)CCCC(C)(C)C1 c1(C(=O)NC(N2CC(C(=O)NCC(C)(O)CN(C)C)C2)=O)cc(C(F)F)cc(F)c1 C(=O)(CC(C)(C(F)(F)F)Nc1cc(OC)c(Cl)cc1Br)OC C(CCCC(=O)NC(C)CCC1CCCC1)NC(C(C1CC1)SC)=O C1(CNC(CC(=C)C)=O)CCC2(CCN(C(=O)C(CC(C)(C)C)OC)CC2)O1 CC(C)CCC(C(=O)Nc1cccc(N(C)C)c1)NC(=O)C(C)C1(O)CCC1 c1(-c2cn(CC)nc2)cnc2ncc(C(=O)NC(c3ccno3)C)n2c1 c1(C(N2CCC(C(F)(F)F)C2)=O)nnc2ccc(-c3cnccn3)cn12 S(=O)(=O)(c1cccc(C(=O)NC2CC2NC(C2CCC2C(N)=O)=O)c1)N(C)C.NC N1(C(C(C)(C)OCCC)=O)CC2(C)CC1(C(=O)NCc1ncc(C)cn1)C2 N1(C(C(=O)NC(CC)(C)C)CCC2(C)CC2)CCCC(C(=O)OC)(OC)C1 C(c1ccc(C)cn1)=CC(=O)NCC(CCNC(C1C(COC)C1)=O)O N1(C(c2ccc(CC)cc2)=O)CCCC2(NC(C34COC(CCO3)C4)=O)CC2C1 C1(C(=O)NCC(c2noc(=O)n2C)C)CCN(C(C23CC(F)(C2)C3)=O)C12CCC2 CCCC(CC)C(=O)N1CCC=C(CNC(=O)C2=NNC(=O)C2)C1 c1(-c2ccc(CN(C3CCNC3=O)C)cc2)ccc2c(c1)OCC2 c1(NC(C(N2C(CNC(c3c(CC)nn[nH]3)=O)CC2)=O)C)ccc(Cl)cc1Cl c1(C(=O)NC2(C)CCN(C(CCC(=C)Cl)=O)C2)cc(F)ccc1O c1(C(=O)NC(CC2CN(C(c3n[nH]c(C)c3C)=O)C2)C)cccc2c1C(=O)NC2 c1(C(C(N2CC3CCN(C(C4CCC4)=O)C3C2)=O)(F)F)ccc([N+](=O)[O-])cc1Cl C1(NC(C(C)=CC)=O)CC2(C1)CN(C(=O)C(C)SCC1CCCO1)C2 N(C1c2ccccc2CC1C)C(=O)NCc1cc2cc(C)ncc2cc1 C(=O)(C1=CC2CCCCC12)N1CCC(NC(CN(C(C)C)C)=O)C(O)C1 N1(C(CNC(C(CC)C)=O)=O)CCCC(F)(CNC(=O)C(C)(C)C2CCC2)C1 Cc1c(N)ccc(C(=O)NC2CCC(CNC(=O)C(C)(C)C(C)C)C2)c1F c1(C(C(=O)NC(CC)(C)C)N(N2CCCC2)C)ccc(OCC(N)=O)cc1 c1(-c2cc(C(=O)NCC3C(NC(C(CSC)O)=O)CC3)n[nH]2)ccc(C)cc1 c1(N2CC(C)C(F)C2)cccc(S(=O)(=O)NCC(c2ccnn2C)N(C)C)n1 N1(C(C2(CCCC)CCC2)=O)CCCC(CNC(c2cc[n+]([O-])cc2)=O)CC1 c1(CN(C(CCN(C(=O)CC2CCCC2C)CC)=O)C)cccnn1 Cc1cc(Cl)ccc1C(N1CC(CNC(c2c(C)nnn2C(C)C)=O)C(C)C1)=O S(=O)(=O)(c1c(Cl)cc(Br)cc1Cl)N1C2CC(NC(c3cncc(F)c3)=O)C(C2)C1 CC1(C)CC(NC(c2cnn[nH]2)=O)CN(C(=O)C(=Cc2c[nH]cn2)F)C1 c1(NC2CC(NC(C(C)O)=O)C2)ncnc2cc(C(C)(C)C)sc12 C(=O)(CC(C)C(C)(C)NC(=O)C(C)c1cc[nH]n1)Nc1c(CC)nc(C)cc1 N1(C(C2N(C(C)=O)CC(O)C2)=O)CCN(C(=O)CC(C)C)C(C#N)C1 N1(C(C(CNC(CCOC)=O)(F)C(C)C)=O)CCCC2C(=O)NCC12 C1(C(N2CC(COC)C2)=O)CN(C(=O)CCc2cnoc2)CC1C1CC1 O=C(CCCOCC1(CNC(=O)CNC(c2cccnc2)=O)CC1)OC CC1(C)CC(C(N2CCCC(F)(CNC(C3CCC(=O)N3)=O)C2)=O)CC(C)(C)C1 N1(C(C2N(C)CCCC2)=O)CCC(F)(F)C(N=c2nc[nH]cc2C#N)C1 N=c1ncc(C(=O)NCC2CN(C(=O)CC3CCCCCO3)CCO2)c[nH]1 N1(C(C2(C)C(C)CN(C(=O)C(C3CCCCC3)F)C2)=O)Cc2cccnc2C1 C(=O)(C1=CCCSC1)NC(C(=O)NC1CCN(CC)CC1)Cn1cncn1 c1(C(=O)NC2CCN(C(C(CC)(C#N)CC)=O)CC2O)cccc(P(C)(C)=O)c1 C1(C)(C(N(C(CCC)C)CC)=O)CCCN(Cc2ccc(N)c(Cl)c2)C1 c1(C(=O)NC2CC(CNC(C(C)=CC)=O)C2)cc(CS(C)(=O)=O)oc1C c1(C(N2C3CC(NC(C(c4ccccc4)C)=O)C3CC2)=O)cc(Cl)c(F)c(Cl)c1 N1(C(CC(=O)OC(C)(C)C)=O)CCC(C(N2CCC2(C)C)=O)(CF)C1 C#CCCCC(C)C(=O)N1CCN(C(=O)Cc2cccc(C#N)c2)CC1COC CC(C)(C)CCC(=O)N1CCCC(CNC(c2n[nH]cc2F)=O)C1 CC(C)C(C)(CNC(=O)C#CC1CC1)NC(=O)Cc1ccc(-n2ccnc2)cc1 C(=O)(C(C)S(=O)(=O)C(C)C)N(CCOC)CCNC(c1c[nH]cc(C)c1=O)=O c1(OC)ccc(CN2CC3CCN(Cc4ncc[nH]4)C3C2)c(F)c1F C=CCC(C)C(=O)N(C1CC(C#N)C1)CC(=O)NC1(CC(=O)OC)CC1 CC1CCC(CNC(=O)Cc2cc(O)nnc2O)N(C(c2ccncc2)=O)C1 N1(C(C(CCOC)SC)=O)C(CC(=O)N(C(C)COC)CC)C2CCCC12 CC1(C)CCCC1C(=O)NCC1CCC1NC(=O)CSc1cccc[n+]1[O-] C1(NC(Cc2c(C)nc(C)s2)=O)C(C)CCN(C(=O)CNc2ncccn2)C1C c1(C(=O)NCC(F)CNC(=O)C(F)CC2CCCC2)noc2c1CCCC2 c1(C(=O)NCCC(=O)Nc2c(C)cccc2)n[nH]c2c1CCC(=O)C2 C1(C(=O)NCC(CC)C)CC(N=[N+]=[N-])CN1C(c1cc2occc2[nH]1)=O c1(C(=O)NCC2CC2C(=O)NC2(CCO)CCC2)ccnc(-n2cccc2)c1 c1(C(=O)NC2C(CNC(=O)C=CC=C(Cl)Cl)CC2)cc2nc[nH]c2cc1F c1(-c2cn(CCNC(C(C)NC(c3ccc(C)o3)=O)CO)nn2)ccc(=O)oc1 C1(NC(c2cncc(SC)c2)=O)CC(CNC(c2nnn(C)c2C)=O)C12CCC2 C(CS(=O)(=O)CC(=O)NCC(C1CCCC1)NC(=O)C(C)O)OC C(CCN(C(=O)C(C(C)C)NS(N)(=O)=O)C)(C(C)C)NC(Cc1nc(C)sc1)=O C1(CNC(C(=O)NC(c2ncnn2C)C)=O)CCC2(CCCC2)O1 CCS(=O)(=O)NC(C)C(=O)N(C1CC(NC(C2(OC(C)=O)CC2)=O)C1)C n1(CC(N2C(CNC(COC)=O)C=CC2)=O)c(C(C)C)nc2ccccc12 CC1CCCN(C(=O)C(c2cccs2)NC(c2ncn3c2CCC3)=O)CC1 c1(OC)nc(C)ncc1NC(c1cncc(NC(=O)Cc2cscn2)c1)=O c1(NC(C)Cn2c(N(C)C)nnc2CCCS(N)(=O)=O)ccc([N+](=O)[O-])cc1 c1(C(=O)NC2C(NC(C3CC(CCC)C3)=O)COC2)c(NC(C)=O)c[nH]c1C N1(C(CC)=O)CCC(C(F)CNC(C2CCCN2C)=O)CC1 C1(OC)C2CN(C(=O)Cn3cc(C(c4ccc(F)cc4)O)nn3)CC12 c1(CNC(=O)NCC2CCCC23CC3)ccccc1-c1cncnc1 CC1CCC(F)(C(=O)NCc2ccccc2CN(C)C(c2c[nH]c(=N)s2)=O)CC1 C1(CC)(CC)CC2CN1C(=O)CCCn1cc(nn1)CN2.C(=O)(CC(C)C)NC CC1C(=O)NC(=O)CN1C(C12CCN(C(c3ccc(N)cn3)=O)CCC1C2)=O C1(C(N(C)CC2(O)CCOC2)=O)CN(C(=O)CCS(C)(=O)=O)CC(C)(C)C1 c1(NCC2(CNC(C=CCOC)=O)CCC2)ncnc2sc3c(c12)CCC(C)C3 N1(C(C2C(NC(C3N(C)CC4(CC4)C3)=O)CC2)=O)CCC12CCSCC2 c1(C(=O)OC)ccc(C(N2CCC(NC(=O)C(C)OC)C2)=O)cc1[N+](=O)[O-] CC1CN(C(=O)C(C2CCOCC2)O)CCN1C(=O)C=CC1CCCN1C n1(CC(=O)NC(C(CO)NC(C(n2ncc(C)c2)C)=O)C)ncn(C)c1=O c1(C(=O)NCC(C2CCC2)NC(=O)CNC(c2ccco2)=O)ncc(Cl)cc1F C(c1ccc(C)cc1C)=CC(=O)NCC1(F)CCC(CNC(C(CC#C)C)=O)C1 C1(NC(C2(C)CCC(C)CC2)=O)CCC2CC1CN2C(c1ncnc(O)c1Br)=O C1(CNC(c2ccc(C)cc2)=O)CC(NC(c2cc(Cl)cnc2O)=O)C12CCC2 c1(CC)cccc(C(=O)NCC(C)CN(C)C(C2CN3CCC2CC3)=O)c1F c1(SC)cccc(C(=O)NC2CCOCC2NC(=O)C(c2ccncc2C)C)c1 Cn1ncc2cc(C(N3CC=CC(NC(c4cnccn4)=O)C3)=O)sc12 c1(CNC(=O)CSCCNC(C2CCOC2C2CC2)=O)ccc(F)cc1F C(CCS(C)=O)(C(=O)NCC1CCC1NC(=O)C=Cc1ccccc1F)N(C)C N1(C(C2(OC)CCOC2)=O)CC(n2cc(-c3cccc(F)c3)nn2)C(C)C1 CC(C(=O)N1CCCC(CN(C(=O)Cn2nnnc2C2CC2)C)C1)P(C)(C)=O C1(NC(C2C3CCN(C(C4CCOC4)=O)C23)=O)CC(C2CCCC2)C1 c1(C(N2CCC(C)(CNC(C3(CO)CC3)=O)CC2)=O)c(F)ccc2n[nH]cc12 C1(NC(=O)NC(C)CCc2cn[nH]c2)CN(C(=O)CN(C)C)CCC1(C)C C1(C)(C(N2CC3C(NC(c4c(COC)cc[nH]4)=O)C3C2)=O)CCC2CC2C1 C#Cc1ccc(C(=O)NCCCN(C(C2CCCSC2)=O)C(C)C)nc1 N1(C(C2C3CN(C(c4ccc(SCC)cc4)=O)C2C3)=O)CC2C(C1)C2(C)C C=CC1(CC(=O)NCCC2CCCCN2C(C2CCCC2(F)F)=O)CCCCC1 C1(CNC(c2ccc(CO)c(F)c2)=O)CC2CCC1N(C(c1csc(Cl)c1)=O)C2 c1(OCCC)ccc(CCC(=O)NCC2CCN2C(C2CC(F)C2)=O)cc1 c1(CNC(C2(CNC(C(C)n3cncn3)=O)CCC2)=O)ccc(F)cn1 N1(C(C2(C)CC(O)CN2C(C2CCC2C#N)=O)=O)CCC2(CNC(=O)C2)C1 N1(C(C(C)(C)n2cnnn2)=O)CCC(C(=O)NC(C2CC2C(=O)OC)C)=C(F)C1 Cc1ccc(F)c(C(=O)NCC2CN(C(c3cc(C(C)(C)C)no3)=O)CCO2)c1 c1(C(N2CC(NC(C(C)CO)=O)C(c3cnn(C)c3)C2)=O)ccn2ccnc2n1 C#CCCCCCC(=O)N1CCCC(C(=O)NCCc2cccc(O)n2)C1C c1(OCC)ncc(C(=O)N(CC(C)(C)CNC(=O)CC#N)C)cn1 Cc1ccc(S(=O)(=O)N2CCC(C(N3CC(N(C)C(C)C)C3)=O)CC2)cc1C CN1CCN(C(=O)COCCNC(=O)CC2CCOC2(C)C)C(CCO)C1 c1(C(N2CCC(c3cn(CCNC(C(C)C)=O)nn3)C2)=O)cnc(O)nc1O CC1(O)CC(C(=O)NC(C2CCCCC2)CNC(=O)C2CC2)C1 N1(C(Cc2cc(C)cc(F)c2)=O)CCC2CN(C(c3n[nH]cc3C)=O)CC12 C(=O)(CCC(F)(F)F)NC1(C(N(C)CCc2cccnc2)=O)CCC1 N1(C(c2cn(C)nc2C(F)(F)F)=O)C2CCC1C(NC(=O)C1CC1)C2 c1(-c2cn(CCNC(C3C(F)(C(=O)OC)C3)=O)nn2)cc2ccccc2s1 Cc1cnn(C(C)C)c1C(=O)NCC1CN(C(C2CC(C)(F)C2)=O)CC1O Cc1nn(C)c(C)c1C(=O)NCC1COCC1NC(=O)Cc1cc(F)ccc1O n1(CC)cnc2[nH]c(=NCCNS(C)(=O)=O)nc(N3CCC4(C)C(C3)C4(Cl)Cl)c12 c1(C(=O)NCC2CN(C(CCc3cc(C)no3)=O)C(C)C2)ccc(Cl)c(N)c1 C1(NCCn2c(C)cc(C(=O)O)n2)CC(C2CCC2)C1 C1(NC(c2ccn(C)n2)=O)(CO)CCCN(C(=O)Cn2cccc(N)c2=O)C1 c1(CCC(=O)NC2N(C(C(C)SCC(=O)NCC3CCCO3)=O)CC2)nc(O)n[nH]1 c1(OC)cc(C(=O)NC(CNC(=O)C(N2CCC(C)C2)=O)C2CCC2)cc(C)n1 C=CCCCC(C)(C)C(=O)N(CCNC(c1ccc(C(=O)NC2CC2)cc1)=O)CC c1(C(=O)NC2(CC)CN(C(c3csnc3OC)=O)C2)cc(C)c(F)c(C)c1 Cc1cc(C)c(C(N2CCN(C(=O)Cc3occc3C)CC2C)=O)cc1Br C1(CNC(c2n(CCOC)nnn2)c2cnc(Cl)s2)CC2CC1CC2O C1(NC(=O)C(Cl)=CCl)CC2CC1CN2C(c1cc(C(F)(F)F)cc(O)n1)=O N1(c2n(CCCOC)c(-c3c[nH]cc3C(F)(F)F)nn2)CC2CC(F)(F)C2C1 C1(c2nnnn2CCCSC)(NCc2cnc(CC)o2)CCOCC1C C1(CC)CN(C(=O)CC2OCCO2)CC1C(=O)NCC(C)(O)C(F)F CCCC(O)C(=O)NC1(COC)CCN(C(c2ccnc(-n3cccc3)c2)=O)C1 CCCC(CNC(c1ccsn1)=O)NC(=O)Cc1cnc(C)[nH]1 CC1CCc2nc(NC(=O)CSc3nnc4n3CCNC4=O)c(C#N)cc2C1 S(=O)(=O)(c1cc(Br)ccc1Cl)NC1CCC(CC(N2CC(O)C(F)C2)=O)CC1 C1(NC(c2c(OC)nccn2)=O)CN(C(C2CC2(C)C)=O)CC(F)(F)C1 C#CCC(C)(C(=O)NC1COCC1N=[N+]=[N-])NC(=O)CCOCC(F)F N1(C(CSC(C)C)=O)CC2CN(CCc3ccc(OC(F)F)cc3)CC2C1 C12CCCC1C(=O)N2.C1(COCC)(NC(=O)C2CC2)CCC1 CCC(CC(=O)N1CCN(C(=O)CCC=CC(C)C)C(C2CCC2)C1)C(F)F c1(C(=O)NCCCOCCC(N2C(C)(C)C(O)CC2)=O)c[nH]c2cnccc12 C=CC1CCCN(C(=O)CCC(C)NC(=O)CN2CC3CC3C2)C1 C1(CC(=O)NCC(C)N(C(COCCC=C)=O)CC)CCCOC1 N1(C(C2(CC#C)CC2)=O)C2CCC1CC(NC(c1csc(C)c1C)=O)C2 C1(NC(CC2CC(SC)C2)=O)CC2(C1)CC2NC(c1cc(C)no1)=O Cc1cnn(C)c1CC(=O)NC1CN(C(c2cscc2C(F)F)=O)CC1O N1(C(C2CN(C(C)C)C(=O)C2)=O)CCN(Cc2cc(O)c(O)cc2O)CC1C#N N1(C(C2CCCCC2)=O)CCCC(Cn2cc(CN3CCOCC3)nn2)C1 c1(NS(CC(C2CC(F)(F)C2)OC)(=O)=O)ncc(C)cc1Br CC1CCc2ccccc2N1CCNC(N1CCN(C(N)=O)c2ccccc21)=O C12(C(=O)NCC(C)N(C(=O)Cc3cccn3C)CC)CCCC1OCC2 C1(NC(COC)=O)CN(C(c2cccc(-c3cccc(C)c3)c2)=O)CC1(C)C C1(O)(CC(=O)NC(CNC(CSCCC)=O)C2CC2)CCC1 C(=O)(C1=CC(O)CCC1)NC1CC(NC(C(C)(C)Nc2ccccn2)=O)C1 c1(NC)cnc(C(=O)NCC2(C(=O)NC3CCCC3CCO)CCC2)cn1 C1(C(N2CC(OCCNC(c3coc(O)n3)=O)C2)=O)CCC2(CCC2)C1 c1(CC)[nH]nc(Cl)c1C(=O)NC1CCC1NC(=O)C(CC1CCCCC1)OC c1(CC(=O)N(C)CC2N(C(C(C(C)C)SC)=O)CCCC2)cccc2c1OCO2 S(=O)(=O)(c1cc(NCCNC(=O)Cc2csnn2)ccc1F)N(C)C S(=O)(=O)(c1c[nH]c(-c2nccn2C2CCN(c3ccccc3Cl)C2)c1)NC(C)C c1(C(N2CC(NC(C3CCCCC3(F)F)=O)(CO)C2)=O)n[nH]c2c(F)cccc12 N1(C(C(=O)Nc2ccc(CC)cc2C)C)CCCCCCC1C C1(C(=O)NCCCOCCNC(=O)C(F)(F)c2ncccn2)CCCCC1 C1(C(=O)NC2CCC(C(=O)NC(CC(=O)OCC)C)C2)CCCCC(=O)N1 C1(CNC(Cc2cc(C)on2)=O)CCN(C(c2cc(Br)c(C)o2)=O)CC1 C(=O)(C1=NOC(C)C1C)NC(CC=C)CNC(c1csc2nnsc12)=O C1(CC)CCC(C)CN1C(C1(CNC(=O)Cc2cc[nH]c2)CC(C)(C)C1)=O C(=O)(CCCCC1CC1)N(C(C)C(=O)N(C(C)C(C)C)C)CC C1(O)(C(N(C(CC(N2CCC(N(C)CC)C2)=O)C)C)=O)CCCCC1 C=CCCCC(C)(C)C(=O)N1CC(C2(NC(=O)C(C)CC(=O)OC(C)(C)C)CC2)C1 C(=O)(C(F)CC(C)C)N1CCC(CCNC(CCN2CCN(CC)CC2)=O)C1 C1(NC(C=COCC)=O)CN(C(=O)C=C2CCCC2)CCC1c1cccc(F)c1 C1(CC(=O)NCC2CC(NC(c3cc(C)sc3)=O)C2)CC(=O)NC1=O Cc1cc(C(N2CC(CNC(c3cncn(C)c3=O)=O)CC2C)=O)ccc1O C(=O)(C(C(C)(C)C)N(C)C)N1C(CCNC(c2c(C(C)C)cco2)=O)CCC1 N1(C(c2nn(CC)c(C)c2)=O)CCN(C(=O)Cn2cc(Br)c(=N)[nH]2)C(C)C1C CC(C)C(O)C(C)(C)C(=O)NC1CN(C(=O)C=CCN2CCCCC2)CC1C C(=O)(C1COc2ccc(F)cc21)N1CC(O)(C(C)NC(=O)Cc2ccoc2)C1 c1(CC(=O)NCCN(C(=O)CC2CCC2(C)C)CC)ccccc1C N1(C(CSC(C)(C)C)=O)CCC(O)(CNC(=O)CC2CC=CCC2)C1 Cc1ccc(CCC(=O)N(C2CCNCC23CC3)Cc2cn(C)cn2)c(C)n1 CCC(C)C(O)C(=O)N1CC(C(C)(C)O)(CNC(=O)CCc2ccco2)C1 Cc1cc(C(=O)NC23CC2CN(C(=O)CCC2CCCN(C)C2)C3)c(C)c(C)c1 c1(SCC)cc(C(=O)NC2CSC(C)C2)ccn1 CCC(O)C(F)(F)C(=O)N1CCCC(CC(=O)NC2CCN(C(C)C)CC2)CC1 Cc1nnc2ccc(C(=O)NC3CCCC(NC(=O)CCC4CC4)CC3)cn12 Cc1ccc(OCC(=O)NC(C(=O)NCc2[nH]nnc2C)c2cccs2)c(C)c1 C1(C(C(=O)OCCC2(C(F)(F)F)CCC2)F)CCOCC1 c1(CC)cc(C(N2CCCCC2C2CCN(C(=O)C(C)(C)CO)CC2)=O)ccn1 CC1OCCN(C(c2csnn2)=O)C1C(=O)NC1CCC(C2CC2)C1 C1(C(=O)NCC2(O)CCC2)(NC(=O)Cc2ccc[nH]2)CC(CO)C1 Cc1cc(C(N2CCC(N(C)C(C3COC3)=O)CC2)=O)ccc1-c1ccccc1 N1(C(CC2N(C(COC3(C)CCC3)=O)C3C2CCC3)=O)CC2CC(O)CC2C1 Cc1cc(N2CCC(O)C2)ccn1.c12ccccc1CN(C1CC3CNC1C3)C2=O c1(CC)ccc(CCC(=O)NC(C2CN(C(=O)C(C)CSC(F)(F)F)C2)C)cc1 C(=O)(CC(C)C(C)(C)NC(=O)CN(C)C(=O)OC)N1CCC(O)(CCC)CC1 c1(NCCC(C)(C)CO)ccc(S(=O)(=O)NCc2ccsc2Br)cc1F C12(CNC(=O)CC3CCC3)COC(CNC(c3cccc(CC(F)(F)F)c3)=O)(C1)C2 c1(C(N2C(C)CCC(NC(=O)C(F)(F)CC3CC3)C2)=O)ccc2oc(O)nc2n1 CC1CCCCC1C(N1CCC(C(C)(C)CNC(=O)C(F)=CCCF)CC1)=O CCC(CC)(CCO)NC(=O)N(C1CC1)CC1CCCC1(C)C Cc1ncn(C)c1C(C)NC(c1nnnn1C)C C1(CNC(C2C3CC3CN2C(C2CC3CCC3C2)=O)=O)(CO)CC2CC2C1 CC(C)CC(O)C(=O)NC1CCCC1N1CCN(C(c2cscc2SC)=O)CC1 CC(C)C(C#N)C(=O)NCC=CC(=O)NC(c1ccco1)C N1(C(CCC)=O)CCCC(C)(NC(c2ccnc(OC)c2)=O)C1 C(c1cc(F)c(F)c(F)c1)=CC(=O)NCC1CC(CNC(C2CCC2)=O)CO1 C1(CNC(CCCOC)=O)CC(NC(=O)CCn2nc(C)nc2C)C1(C)C C(C1CCCCCC1)=CC(=O)NC1(CC)CN(C(=O)CC2CCCC23CC3)C1 C1(C(=O)NCC2CC(NC(c3sccc3C(F)F)=O)C2)COCCO1 C(=O)(C(CC)CC(F)(F)F)NC(CC)CNC(=O)C(C)Cc1ccccc1Cl CN(S(=O)(=O)N=S(C)(=O)C(C)(C)C)Cc1cccs1 N1(C(CCc2n(C)ncc2)=O)CCC(NC(=O)C=CCO)CC1C1CC1 c1(CC(=O)NC2(C)CC(NC(c3c(C)oc(C)c3C)=O)C2)ccc2n[nH]cc2c1 c1(CCC(=O)NC23C(CN(C(C(C)OC)=O)C2)C3)cc(F)cc(F)c1 c1(CN2CCN(CCCNC(CC(C)(C)C)=O)CC2)c[nH]c2cccc(Cl)c12 c1(CCC(=O)N(C2CCN(C(C3CC4CC4C3)=O)C2)CC)scnc1C C1(C(N(CCOCC)C)=O)CC(C)CCN1C(c1cc(C)[nH]c1C)=O N1(C(C2CN(C)C2)=O)CC2(CNC(c3ccc(F)c(F)c3N)=O)CC1CCO2 N1(C(c2c(C)con2)=O)CCOCC(CNC(C2CCCCN2S(C)(=O)=O)=O)C1 C1(C(=O)NCCCNC(C(C(C)C)Cc2ccccc2)=O)COCC2(CCC2)O1 C(=O)(C(O)C(F)(F)F)NC(C(=O)NCC1CCCSC1)Cn1cccn1 c1(C(N2CCC(C(C)C(=O)NC3CC4(CCC4)C3)C2)=O)ccc2ccoc2c1 C(CO)(C(C)(C)CO)NC(C(C)(N(C)C(C1CC12CC2)=O)C1CC1)=O C1(C(N(CCN(C(C(C)=C(CC)C)=O)C(C)C)C)=O)CCCCC1F c1(C(=O)NC23CC2CN(C(=O)CNc2ncccn2)C3)ccc2ncsc2c1 C1(C(=O)NCCCC(CCC)NC(=O)CCCC(F)F)CCS(=O)(=O)C1(C)C CC1(C)C(C(N2CC(F)CC2CNC(C2(O)CCOCC2)=O)=O)CCS1(=O)=O C=CCC(CC(C)C)C(=O)NC1CCCC1NC(c1cnc(C(=O)OC)s1)=O C1(NC(CC(=C)C)=O)CN(C(C2CC23CCOCC3)=O)C2(CCCCCC2)C1 c1(C(=O)NC(CCNC(C(CC)F)=O)(C)C)ccc2cc([N+](=O)[O-])ccc2n1 C(=O)(CC(F)(F)C(F)F)NC(CNC(c1ccc(CC)cc1N)=O)(C)CC(C)C n1(CC(N2CCC(NC(Cc3c(C)non3)=O)C2)=O)c(=O)oc2ccccc12 C1(CC(=O)NCCC(C)NC(=O)C(C)N(C)C)SC(=N)NC1=O C(=O)(CC1=CCOCC1)NCC1N(C(CC(C=C)(C)C)=O)CCCC1C C1(CNC(CCc2c(C)noc2C)=O)N(C(=O)CC2CCC(=O)O2)CCC1(C)C c1(C(N2CCCC(NC(c3ncc(NC)nc3)=O)C2)=O)c(F)cccc1Br c1(SC(C)C(=O)N(C2CCN(C(C3(C(F)(F)F)CC3)=O)C2)C)ccccc1 Cc1csc2cc(C(=O)NCC3(O)CCN(C(c4ccc(F)cc4F)=O)C3)[nH]c12 c1(C(=O)OC)cc(C2(C(=O)NCCOCCOCCNC(C)=O)CCCC2)[nH]n1 C1(NC(C(C)CC2CCCCC2)=O)CC2CCC1N(C(=O)CCCC(C)(C)C)C2 c1(C(N(C2CCN(C(=O)CCC#N)C2)C)=O)ccc(C2CC2)c(Cl)c1 N1(C(C=C(C)C(C)(C)C)=O)CCC(C)C(N(C)C(C2CCC3(CCC3)O2)=O)C1 c1(C(N(C(C)CNC(=O)Cc2cnccc2Cl)C)=O)cc2n(n1)CCN(C)C2 C1(OC)CC(NC(=O)C(F)(F)C(F)F)CN(C(=O)CC(O)c2ccccc2)C1 Cc1cc(CN2CCC(N(C)C(c3c(Br)cnn3C)=O)C2)c(C)cc1Br C(=O)(N=c1ccn(C)[nH]1)C1(NC(c2c(CC)ncs2)=O)CC(O)C1 Cc1ccc(C(=O)NCC2CN(C(=O)CSCC(N)=O)CCO2)c(N)c1 c1(C(N2CC(C)(C(=O)Nc3ccc(C)cc3Cl)C2)=O)ccc(Cl)c(S(N)(=O)=O)c1 O=C1CCCCC(C(=O)NCCC2CN(C(c3ccncc3)=O)C2)N1 C(=O)(CS(=O)(=O)NC(C)(C)C)NCC(C)NC(=O)C(N1CCOCC1)C S(=O)(=O)(c1ccc(Br)s1)N1CCN(CC(=O)N(C2CC2)Cc2cccnc2)CC1 C(C)(CCCCCO)NC(C1(CNC(=O)COC2CCCC2)CC(=C)C1)=O c1(C(=O)NCCN(C(=O)C#CC2CC2)CCCN(C)C)ccc(OCC(N)=O)cc1 N1(C(C(C(C)C)O)=O)C(CNC(c2c[nH]c(C(N)=O)c2)=O)CC2CCCCC12 Cn1c(C(=O)NC2CC2NC(=O)Cc2csc3ccccc23)cc2sccc12 N1(C(C(N)=O)=O)CC(NC(C2CCN(C(C3CCC3)=O)CC2)=O)C(CC2CC2)C1 c1(C(N(CC)CC2CCCN(C(=O)C(C)C3CCCC3)C2)=O)nn(C)c(N)c1C C1(C(N(C2CCN(C(c3sccc3-n3ccnn3)=O)C2)C)=O)CCC(O)C1 c1(CC)c[nH]c(=NCCc2ccc(C(=O)OCCOC)cc2)o1 Cn1nnc2cncc(C(N3CC(C)(NC(C4CCC5CCCCN45)=O)C3)=O)c12 C1(c2nnnn2C2CCCC2)(NC(C)Cc2ccccc2Br)CC(C)SC(C)C1 c1(C(=O)NC2C(NC(c3cccc(C(=O)NC)c3)=O)C2)cccc2sncc12 N1(C(CC(=O)N(C)C)=O)CCN(C(=O)CCc2nc[nH]n2)C2CCCCC12 c1(C(=O)NC2(C)CCN(C(CCCC#C)=O)C2)ccc(F)cc1C Cc1cc(Cl)nc(NC(c2cccn2Cc2cccnc2)=O)n1 c1(OC)cncc(C(=O)NCC2CCCCCN2C(c2n[nH]c(C)c2Cl)=O)c1C c1(C(C)C)ccc(C(=O)NCCC(O)CNC(C2CNC(=O)C2)=O)c(O)n1 C(C)(C(=O)NCCOc1ccncc1)(N(C(C=CC(=O)N(C)C)=O)C)C1CC1 c1(C(=O)NC(COCC)C)coc(CNC(c2ccc(C(N)=O)[nH]2)=O)c1 C1(CNC(C(C(C)(C)C)(C)C)=O)CC2(CCN(C(C3CCNC3=O)=O)CC2)CO1 N1(C(C2(CC=C)CCCC2)=O)CCCC(N(CCO)C(c2ccc(C)s2)=O)C1 Cc1cccc(C(=O)NC(C)(C)C(C)NC(c2ccc(Cl)s2)=O)c1F N1(C(CCc2ccc(C)nc2)=O)CCN(C(c2cc(C)no2)=O)C2CCC12 N1(C(C2C(C)(Br)C2)=O)CCC(C2CCN(C(C3CC34CCC4)=O)CC2)CC1 S(=O)(=O)(c1cnn2ccc(=NCCC(F)F)[nH]c12)N1CCC(C(C)C)C1 c1(CC)ccc(C(=O)NC2CC(O)C2CC(=O)N(C)Cc2cnc(C)s2)o1 Cc1ccc(C(C)C(=O)NCC2CC(NC(=O)CN(C3CCSC3)C)C2)s1 C(=O)(C1CCc2cc(Br)ccc21)N1CCN(C(C(COC)C)=O)CC2(C1)CC2 N1(C(CCC(C)SC)=O)CC(C)OC2(CCN(C(c3cc(C(C)C)no3)=O)C2)C1 c1(N2CCCC(n3c(O)ncc3)C2)nccc(=NCC#CC2CC2)[nH]1 c1(CN2CCCC2)c(F)cccc1F.c12nnc(o1)CC1N(CC1)C2C CCC(C)(C#N)C(=O)NCCC1CCCN(C(c2csc(COC)n2)=O)C1 Cc1c(CC(N2CCCC2C2(NC(=O)C(C)NC(N)=O)CC2)=O)cnn1C Cn1cc(C(=O)NCCCS(=O)(=O)N2CCCC2)c(Br)n1 c1(C(=O)NCC(C)N(C(=O)C(N2CCOCC2)C2CC2)C)ncoc1C1CCC1 C1(C(N(CC(=O)OCC)CC=C)=O)CCOCC1NC(c1cccc(=O)o1)=O N1(C(C2(OC)CCSCC2)=O)CCC2(C1)CN(C(C1CC(C)OC1=O)=O)C2 c1(OC)ccc(C)c(OC)c1C(N1CC(NC(c2cc(F)c[nH]2)=O)CC(F)C1)=O C(=O)(C(CC(C)CC)NC(C1C=CC=CC=C1)=O)NCCCCC#CC C12(CNC(COC)C(=O)NCC(C)N(C)C)CCCC(CO1)C2 C1(CCC)CN(C(c2ccccc2F)=O)CCN1C(C1CC(C)N(C)C1)=O c1(OC)ccsc1S(=O)(=O)NC(=O)C(C)Oc1ccc(Cl)cc1Cl CC1(C)CC(NC(=O)C(CC2CC2)NC(C2(O)CCSCC2)=O)C(C)(C)O1 C1(CC(=O)N(C2CCCNC2)C2CC2)CNC2CCCCC12 C(=O)(C1=CCCS1)N1C(CN(C(=O)CCOC2COC2)C2CC2)CCC1 C1(C(=O)NCc2nc(C)on2)CN(C(C2CCOC2C(C)C)=O)CCO1 c1(C(=O)OCC=C)c(OC)sc(C)c1C.c12cccc(c1)NC(=O)N2 CC(CN(C)C)CCC(=O)NC1CC1CNC(c1ccncc1)=O C(=O)(N1CCC(C(N2CC(N(C)CC)C2)=O)O1)c1n(C=C)nnc1 C1(C(=O)NCc2ccc(Br)s2)COCCN1Cc1cccc(O)c1 N1(C(C(N2CCNC2=O)C)=O)CCC(CCNC(C2CNC(=O)O2)=O)CC1 CC1(C)CCCCCN1C(=O)CN1CCN(C(c2ccccc2)(C)C)CC1.C(C#N)O c1(N2C(CNC(CNC(C=C(C)C)=O)=O)CCCC2)ncnc2occc12 C1(C(=O)NCCN(C(C=C(C)C(F)F)=O)C(C)C)CCCS(=O)(=O)C1 N1(C(C(COCC)NC(=O)Cn2nccn2)=O)CCCC(C)(COC)C1 C1(CC)C(C(=O)NCC(C(C)(C)C)NC(=O)CSc2nncn2C)CCN1C N1(C(c2cnn(C(C)C)c2)C(=O)NCCCSCC)CCC2(CC(OC)C2)C1 CCC(C)CC(C)CC(C)C(=O)N1CC(c2ccc(Br)cn2)(O)C1 c1(SCCCCN(C(=O)CC(C)O)CCNC(C=C(C)Cl)=O)ccccc1 CC1(C(=O)NCC#CCNC(C23CC2COC3(C)C)=O)CCC(F)(F)CC1 C=CC(C)(CC)C(=O)NC1CN(C(=O)C(c2ccccc2)N(C)CC)CCC1C c1(C(N(CCCC(N2C(COC)COCC2)=O)C)=O)cc(C)c(N)cn1 c1(C(N(C2CC2)Cc2ccc(-c3ccc(CC)s3)cc2)=O)nccn2ccnc12 C(=O)(CC(C)C(C)(C)C)NC1CCC(NC(CCCCC#C)=O)C1 c1(-c2cn(CCCNC(c3nn(C)c(Br)c3)=O)nn2)ccc(O)c([N+](=O)[O-])c1 c1(CNc2ccccc2)ccc2oncc2c1.CC(C)C1CO1 C1(C(N2CCC(N(C(C(CCC)OCC)=O)C)CC2)=O)OCC2CCCCC12 Cc1cccc(C(=O)NCC2CCC2C(=O)NCC2(O)CCC(C)C2)n1 C1(C(=O)NCC2(C#C)CCC2)CC(CC)CCN1C(C1CCC(=O)NC1)=O CC1(C(=O)NCC2(CNC(=O)CCc3ccc(O)cc3)CCCC2)CNC(=O)C1 C(CCCC(=O)NCCOCCCCCNC(=O)CC1CCNC(=O)C1)OCC c1(CC(=O)N(C)CC2(NC(CCOCCN(C)C)=O)CC2)cccnc1Cl c1(SCC(=O)NCC2N(C(CCC3CC(OC)C3)=O)CC2)nc(C)cc(C)n1 C(C(N=[N+]=[N-])C(=O)NCC=CCC(=O)NCCC1CCN(C)C1=O)OCC N1(C(CCC=C(C)C)=O)CC(F)(F)CC1C(N1CCC2(CCC2)C1)=O c1(-c2c(C(=O)NCc3nc(C)sc3)n[nH]c2)cccc2cc[nH]c12 c1(OC)cccc(N2CCCC(CN(C)C(C3CCCC3C)=O)C2)c1[N+](=O)[O-] C=C(C)C(CC(=O)NC(CC(N1CC=CC1(C)CO)=O)C1CC1)OCC N1(C(C(C#C)(C)C)=O)CC2CN(C(=O)C=Cc3ccc(C)s3)CC2(C)C1 CC1OCCN(C(=O)CN(C2CCC2)C(C2CC3(CCC3)C2)=O)C1CO C1(C(=O)NC2C(CSC)CCC2)CCCCCCN1C(c1cc(C(C)C)no1)=O C1(CC(=O)NC2(CC)CC(C)(C)C2)C2CCCC2N1C(C1(COC)CC(=O)C1)=O C(=O)(C1=NN(CC)C(=O)CC1)NCCN(C(=O)Cc1ccc(F)cc1C)CCC C(=O)(C1=NOC2(CCC2)C1)N1CCC(C#C)(C(=O)N(C)CCOC)C1 C1(CC)(CO)CCN(C(=O)C(=O)NC(C2CCOC2)COC)C1 c1(C(=O)OC)c(NC(C2C3CC2N(C(c2csnc2C)=O)C3)=O)sc(C)c1C Cc1cc(C(N2CCCC2C(=O)OC(C)(C)C)C(=O)NC2CCOC2)n[nH]1 C1(NC(C(OC)OC)=O)CN(C(c2ccc(OC(F)(F)Cl)cc2)=O)CCC1CO C1(C(=O)NCC2CC(C(=O)NC3C(C#N)CCC3)C2)CCC(C2CC2)C1 c1(C(C)C)nnsc1C(=O)NC(C)(CNC(C1CCCO1)=O)CO Cc1cccnc1C(=O)NCCC(C)(C)CNC(c1occc1C)=O c1(OC)cnnc(C(N2CCC2C(=O)NCCC2CCC(C)(C)O2)=O)c1 CC(CCSc1ccco1)N=c1[nH]c(N2CCC(=NO)CC2)nc2ccccc12 c1(C(N(C2CCCC2)CC(C)C)=O)ccc2c(c1)CCC2(C)C CCC(CCC(=O)N(CCCC(O)CO)C)NC(c1cn(C)c(=O)cn1)=O C(CC1=CCN(C(C2CCCCO2)=O)CC1)NC(C1CC(F)C(=O)N1)=O N1(C(C=CC=CCC)=O)CCN(C(=O)C(N2CCC(C)C2)=O)CC1C1CC1 c1(C(N(CCN(C(=O)CC2CCCCC2C)CC)CC)=O)nnn(C)c1C C1(OC)COCCN(C(C2CCC(C(C)C)N2C(=O)CCCCC2CC2)=O)C1 c1(OCC)cc(Cl)ccc1C(=O)NC1(C)CCN(CC(C)CC)C1 N1(C(c2cc(C(CC)CC)no2)=O)CCOCC(NC(=O)C(C)=C2CCC2)C1 CC1(C)CN(C(=O)CC23CCCC2C3)CC(CNC(=O)CCC(N)=O)O1 Cc1cccc(C(N2CC=CC(NC(C3COC(C)(C)CO3)=O)C2)=O)c1O C(=O)(C(F)C(C)CNC(=O)C(C)COC)NCCCOCC#C c1(C(=O)NC(C(C)NC(C(CC)F)=O)(C)C)ccc(OC(C)C)c(OC)c1 c1(CN(CC(=O)NC(C)CCNC(C2COCCN2C)=O)C)cccc(C#N)c1 C(C(O)C(CC)CC)NC(CCC1(NC(c2c(CC)cncc2)=O)CCC1)=O C1(NCc2c(N(C)C)cccc2)CN(C(c2cc(Cl)ccc2Cl)=O)CCC1O CC1(C)CC(CNC(c2ccc(F)cc2F)=O)N(C(C2CCCCS2)=O)C1 C1(CNC(C(F)=CCC)=O)N(C(c2ccnn2CCC)=O)CCC1(C)C N1(CC2(C)CCC2)C(=O)CCN(Cc2cccc(-c3ccccc3)c2)C1=O C1(C(NOC(C=C)C)=O)CCN(C(=O)CC)CCC1(C)C CCCCC(CNC(c1c[nH]c(C#N)c1)=O)NC(=O)CSc1cnn(C)c1 C1(NC(C2C(OCC)CC2)=O)C2CCCN(C(=O)CCP(C)(C)=O)C2C1(C)C c1(OC)ccc(-c2ccc(O)c(C)c2)cc1NS(C)(=O)=O.C123CCC(CC1)(C2)N3 C1(CNC(c2csc(CO)n2)=O)COCCN1Cc1ccc(-c2cccnc2)o1 CN=c1[nH]cc(NC(=O)NCCCC2CCN(C)C2)s1 C(C(=O)N(C)CCC1CN(C)C1)(C(C)(C)C)NC(c1c(C)nco1)=O C1(C(N2CC(O)C(O)C2)=O)CN(Cc2cccn2-c2cccnc2)CCC1O C1(CC)CN(C(c2ccn(CCNC(C3C4CC(=O)CC34)=O)c2)=O)CC1O c1(OC(C(=O)NCC2(F)CC(NC(C(CSC)OC)=O)C2)(F)F)ccc(F)cc1 N1(C(c2[nH]c(CC)c(Cl)n2)=O)CCC(NC(c2cc(O)ccc2Cl)=O)C(C)(C)C1 C1(O)(CNC(C(C)Cc2ccccc2Cl)=O)CCCN(C(C2OCCCO2)=O)C1 C1(C(C)NC(C2C(=C)C2)=O)CCN(C(=O)C(C)NC(=O)Cc2cccs2)CC1 c1(C(N2CCC(O)(CNC(C3CC(C)(C)C3)=O)C2)=O)c(Cl)ccc(F)c1F Cc1ccc(O)c(CC(=O)NCCC(C)(C)NC(=O)Cc2ccon2)c1 CCCCC(C(=O)NCC1CCSC1)NC(=O)C(C1CC1)C1CC1 C(=O)(C(C(C)C)NC(=O)CC1CCCOCC1)NCC1N(CCOC)CC1 Cc1nn(CCCN(C)C)c(C)c1S(=O)(=O)NC1COCC1n1ccnc1 C1(CC(=O)NC(C=O)C)CCC(C)(C)O1.C#CC(C)(C)N CC(C)C(C)C(=O)NC(CNC(=O)C(C)OC1COC1)C1CC1 c1(OC)cc(C(=O)OCC(c2cccc(Cl)c2)C)ccc1C#N N1(C(CN(CCC)C)=O)C(CNC(C2C(C)(C)C2(C)C)=O)CCC2CCCCC12 C1(CNC(c2n(CC)ncc2Cl)=O)CCC(C)CN1C(c1ocnc1C1CC1)=O CC(=O)C(C)CC(C)C(=O)N1CCCCC2(CCC2)C1 c1(OCC)ccc(N)c(C(N2CC(F)(F)CC2CNC(=O)C=C2CCCC2)=O)c1 N1(C(C(CCC)OCC)=O)CC(NC(C2CC(C#N)C2)=O)CC2(CCOCC2)C1 c1(C(C)Sc2nnnn2C2CC2)ccc2c(c1)CCO2 C(=O)(C(N)CC(F)F)N(C1CCCC(C)C1)C(C)C1CC1 C(=O)(C1c2c[nH]nc2CN1C(c1cc2n(n1)CCC2)=O)NCC(C1CCCC1)C c1(C(C)(C)CN2CCCC2)nccnc1N1CCCC(Oc2ccccc2Cl)C1 Cc1nn(C)c(C)c1CNC(C1(NC(C2CCCC(=O)C2)=O)CCC1)=O c1(C(=O)NC(CC)CNC(=O)CC2CCCCO2)n[nH]c(C)c1C c1(NC(C(C)(CO)NC(C(CC)OC)=O)=O)cccc(Cl)c1C Cc1cccn2nc(C(=O)NC3CN(C(=O)C(C)(C)C)CCC3C)cc12 c1(C(N2CC(CC(=O)OC)C(C)C2)C(=O)NC2CCCC2)sc(C)c(C)c1C c1(C(N(CCC(C)NC(C2CCOC2)=O)C)=O)c(F)ccc(Cl)c1F c1(C(N2C(C(N3CCC(C)(CO)C3)=O)CCCC2)=O)ccc(F)c(O)c1 c1(C(=O)NC(CSCC)C(=O)NCC23COC(CC)(C2)C3)cncc(C#N)c1 c1(OCC#C)ccc(C(=O)NC2(CNC(C3CCOC(=O)N3)=O)CC2)cc1 C(=O)(C(C)S(=O)(=O)C(C)C)NC1CC(F)(CNC(c2c(OC)ccnc2F)=O)C1 C(=O)(C(C(C)(C)O)NC(=O)C(O)CSC)NCC(CCC)(C)C c1(C(C)C)ncc(C(=O)NCCNC(c2cnc(C(N)=O)s2)=O)n1C Cc1cc(C)n(C(C)C(N2CCCC(CCNC(=O)CCc3cncs3)C2)=O)n1 N1(C(c2c(C)cc[nH]2)=O)CCC2CCC(NC(=O)CC3CN4CCC3CC4)C1C2 CC1(C)C(CC(=O)NCC2(O)CN(C(=O)CCNS(=O)(=O)C(F)(F)F)C2)CC1O c1(C(=O)O)cc(Cl)c(O)c(S(=O)(=O)NCC2CN(Cc3ccc(O)c(O)c3)C2)c1 C(=O)(C1=CNC2=NCCC2=C1)N1CCC(CC)C1CNC(c1occc1C)=O CC(C)CC(C(=O)NC1(C(=O)O)CCN(C)C1)N(C(=O)C(CO)OC)C N1(C(=O)CCC2CCC2)CCC(C2CCCN2C(c2nncs2)=O)CC1 C(C1COc2ccccc21)N(C(C(N)Cc1cccc(Br)c1)=O)CCO CC1(C)CC(CC(N2CCC(O)(CCNC(=O)CNC(N)=O)C2)=O)C(=O)O1 CC1=NNC(=O)C1CC(=O)NC1CN(C(=O)Cc2cccc(O)c2)C1 C1(C(=O)NCC2(C)OCCN(C(C3CC(O)(CC)C3)=O)C2)CCc2nnnn2C1 Cc1nc(C(N2CC3CC3(CNC(=O)CCC(=O)c3cccs3)C2)=O)n(C)n1 c1(NC(CCCC)=O)cc(C)c(S(=O)(=O)N2CCCC2(C)c2cccs2)c(C)c1 C(=O)(C(C)(C)CCC#N)N1CC(CC(=O)NC2(O)CCOCC2)(OC)C1 C=C1CC2(C1)CC(C(=O)NC(C)CNC(=O)CC1CCNC(=O)C1)C2 c1(OC)ccc(CN2CCCC(C)(C(N3CCN(CCCO)CC3)=O)C2)cc1Br Cc1ccn2cc(C(=O)NC3(CNC(=O)C=Cc4cnc[nH]4)CCC3)nc2c1 c1(NC(C(=O)N(CCN(C)C)C(=O)OC)=O)ccc(OC2CCC(C)(C)C2)cc1 N1(C(C=CCN(C)C(c2cc(Cl)n(C)n2)=O)=O)CC(=O)N2CCCC2C1 c1(CC)ccccc1C(=O)N(C1CCC(NC(c2cn(C)cc2C)=O)CC1)C C(C(C)(C)c1ccccc1)(c1nnnn1C)NCCC1CC(OC)C1 C#CCC(C)C(=O)N1CCCCC1CNC(=O)CCNC(=O)CCc1cnco1 C1(NC(C(C)=CC)=O)CCCCC1NC(=O)C=CC1CCCN1C C(=O)(C(C)C1CC1)NC(CN(C(=O)CC1(CSC)CC1)CC)C N1(C(CC2(CC(=O)OC)CC2)=O)CCCC(NC(c2ncn(C(C)(C)C)n2)=O)C1 n1(CC)c(CCNC(c2ccncc2)CC2CCCCC2)nc2ccccc12 c1(-n2ccc(CNC(=O)Nc3c(C)ncnc3)n2)c(F)cccc1F C1(F)(C(=O)NC2CN(C(c3c(C(C)C)cco3)=O)C2)CCS(=O)(=O)C1 c1(OCC(=O)NCC2CN(C(C3C(C#N)C3)=O)C2)cc(F)ccc1Br N(C1CN(C(=O)C(F)C(C)C)Cc2ccccc21)C(C12CC(CCC)(C1)C2)=O c1(C(N2CCC(C)(CCNC(C3CCC(=O)O3)=O)C2)=O)c[nH]c2nccc(Cl)c12 C1(NC(c2nnn(C)n2)=O)CC2CC(C1)CN(C(=O)COc1ccc(O)cc1)C2 CP(C)(=O)CN1CC(C(=O)NCCC2(NC(=O)CCC3CC3)CCC2)C1 N1(C(C(CC[S+](C)C)O)=O)CCCC12CCCN(C(c1ccc(N)cc1F)=O)C2 N1(C(Cc2c(C)ocn2)=O)CCC(NC(=O)CNC(=O)CC(C)C)C(O)C1 c1(C(=O)NC(C(C(C)C)NC(CCC)=O)C)sc2ncccc2c1Cl N1(C(COCCN(C)C)=O)CCCC1CC(=O)NC(C)(C)CNC(=O)CN(C)C C1(NC(C(CCCC)O)=O)CS(=O)(=O)C2CN(C(=O)C3=CCOCC3)CC12 c1(C(C(=O)NCc2cc(CNC(C)=O)on2)O)c(C)cccc1C c1(C(=O)NC(C)(C)CNC(c2n[nH]c(C(C)(C)C)n2)=O)cc2n(n1)CCCC2O c1(C(N2CC3CC2CN3C(C2SCCCS2)=O)=O)c(F)cccc1Cl c1(-c2ncc(C(N3CCC(CC(C)C)CC3)=O)nc2)cc([N+](=O)[O-])ccc1F Cc1c(F)ccc(F)c1C(=O)NC1CN(CC2CCC2)C1.c12ccc(cc1)NC2 CCCCC(O)C(C)C(=O)NC1(CC(=O)NC2CCC3(CC2)N=N3)CCCCC1 Cc1c(C(=O)NCC2CCN(C(=O)CC3CCCCCC3)C2)cnn1CC(C)C N1(C(CCCSC)=O)CCC(NC(c2cc(Cl)nnc2O)=O)C(C)C1 Cc1ccc(C(=O)NCC(C)CNC(C2CCCS(=O)(=O)N2)=O)cc1C(C)(C)C c1(C(c2n(CCCC)nnn2)NCCn2nncc2C)ccc(S(C)=O)cc1 CCCCCCC(C)C(=O)N1CCCCC1CNC(C1CC2COCC2C1)=O C(=O)(C(C)(O)C(C)C)N(CCCN(C)Cc1cc(C)on1)C C1(NC(c2c(C)ccs2)=O)CC=C(C(=O)NCC2CCCS2)C1 C1(NC(C(C)(C)OCC)=O)CCN(C(=O)CCNC(=O)C=CCl)CC1C CC1(C)CCN(C(C2(C)CC2)=O)CC1CNC(c1cncc(C(F)(F)F)n1)=O C(c1cc2ccccc2o1)=CC(=O)NC1CCN(C(=O)Cc2nnc(O)s2)C1 C1(C#N)(C(N(CC(CN(C)C(C2C3CCCOC23)=O)O)C)=O)CCOCC1 C1(NC(C2C(C)=C2)=O)CC1C1CCCN(C(c2cncc(N)n2)=O)C1 N1(C(c2cncc(C#C)c2)=O)CCOC2(CCN(C(=O)CCC=CBr)C2)C1 C1(CCC)CN(C(c2ccon2)=O)CCN1C(=O)CC1CC2CCC(C1)C2 C1(C(=O)NCCN(C(C(C)(C)OCC)=O)C)CNC(=O)CC12CCOC2 c1(C(=O)NCC(C)NC(C(C(CC)C)O)=O)ccc2nc[nH]c2n1 N1(C(CC2(C=C)CCC2)=O)CC2CC(C1)N(C(c1ccc(C#N)[nH]1)=O)C2 CC1CC(CNC(=O)CCC2CCOC2)CCN1C(c1cc[nH]c1)=O C(=O)(C1CCc2nnc(C)n21)NCC(C)NC(C1=C(CC)OCCC1)=O C1(NC(C(N2CCOCC2)C)=O)C=CCN(C(c2ccnc(C3CC3)n2)=O)C1 CC1CN2CCN1C(C(N1CC(CCNC(=O)C(O)CC3CCCCC3)C1)=O)C2 CC(C)(CF)C(=O)NC(CNC(C1(c2ccc(Cl)cc2)CCCC1)=O)C(C)(C)C N(C(=NCC)NCC1(CO)CC2CC2C1)CC(CCC)C N1(C(C(COCC)C)=O)CC2CCC(NC(c3ccn4cccc4c3)=O)(C2)C1 c1(CC)cn2c(n1)CC(C(N1CCC(NC(c3ccc(Br)o3)=O)C(F)C1)=O)CC2 N1(C(=O)OC(C)(C)C)CCCC(F)(CC2CCCCN2CCNc2ccco2)C1 c1(NC(c2ccc(-c3cnc(OC)c(C)c3)nc2C)=O)cc(F)cc2[nH]ccc12 Cn1cc(C(C)(C)C(=O)N2CC(CNC(c3ccoc3Br)=O)C2)cn1 N1(C(C(C)n2cnnn2)=O)CCC(C(=O)NC2CCCCC2C#N)=C(F)C1 c1(C(=O)NCCN(C(CNC(=O)OC)=O)C)cnn(C2CCOCC2)c1 C(CN=C(NCc1cccc(C(C)(C)C)c1)NC1CC1C)NC(C)=O O=C1CN(CC(=O)NCC23CC(NC(c4nccnc4O)=O)(CO2)C3)C(=O)N1 N1(c2nnc(C3CCC(OCC)C3)n2C)CCNC(=O)C1c1ccccc1 C=CCC(CC=C)C(=O)N1CCN(C(=O)C(CC)OCC)C(C)C1 c1(OC)ccnc(C(=O)N(C2CCN(C(=O)CC3C=CCC3)CC2)C)c1N Cc1[nH]c(=N)nc(O)c1CCC(=O)NCC1(CCO)CN(C)C1 Cc1nc(NC2CCC(NC(c3cnn(CCC(F)(F)F)c3)=O)CC2)[nH]c(=N)n1 C1(O)(C(C(=O)N(C(C)CO)C)NC(=O)CP(C)(C)=O)CCCCC1 CC(C)C(C)(C)C(=O)NC12CC1CN(C(C1CC1Sc1ccccc1)=O)C2 C(=O)(CC(C)(C)C(F)(F)F)N1CCC(N(C(=O)CNC(=O)OC(C)(C)C)C)CC1 c1(C(C)=O)ccc(C(=O)NCC(C2CCC2)NC(=O)C(C)c2ccco2)nn1 CCCCCC(=O)NC(CNC(=O)CNC(=O)NC)C1CCC1 c1(C(N(CCN(C(COCCCC)=O)C(C)C)C)=O)cccc(Cl)c1 c1(C(N(C2CN(C(c3ccc(Cl)cc3N)=O)CC2F)C)=O)[nH]cc2c1CCC2 O=[N+]([O-])c1cccc(F)c1CS(=O)(=O)Nc1nccc(N2CCCC2)n1 C=CCCC(N=c1cc(C)[nH]c(=NCC(COC)OC)[nH]1)C1CC1 C1(C(N(CCNC(C2N(C(=O)OC)CCC2)=O)C(C)C)=O)CNC(=O)C(C)(C)C1 c1(C(=O)NCC2OCC(CNC(=O)C=C3CC3)C2)ccnc(N(C)C2CC2)c1 C1(CC(=O)NCC(F)(F)CO)CCC(NC(=O)CC2CCCOC2)CC1 CC(C)C(C)(O)C(=O)NCCC(C)CCNC(c1ccc(C2CCCC2)cc1)=O N1(c2cc(C)ncn2)CCCC(C)(CNC(c2conc2C(C)C)=O)C1 CC1(C)CC(NC(=O)CNC(=O)OC(C)(C)C)CN(C(C23COCC2C3)=O)C1 N1(C(C(C)CC2CCCCC2)=O)CC=C(CNC(C2CCCC3CC23)=O)CC1 CC1CCC(CO)N(C(c2coc(Br)n2)=O)C1 N1(C(C2CN(C)C(=O)N2)=O)CCC(F)C(NC(=O)C=Cc2cccc(Cl)c2)C1 c1(C(=O)NC2CCN(C(CN3CCC(C)CC3)=O)CC2)cnn(C)c1S(C)(=O)=O N1(C(C(C)N(C)C)=O)CCOC2CN(C(c3cnn(C)c3N)=O)CC12 N1(C(C=CC)=O)CCCC2C1CCCCN2C(c1coc(C(C)(C)C)n1)=O C(C)(C(C(=O)N(CCCCO)C)C(C)C)NC(CCC(=O)N(CCC)CCC)=O C1(NC(c2n[nH]c3c2CCC3)=O)CCC2CC1CN2C(c1ccc(Cl)cn1)=O c1(C(=O)NC2CCCC(NC(C3=C(C)OCCS3)=O)C2)c(F)c(F)cc(F)c1F CCC(CCC(=O)NC1(c2cccs2)CC1)NC(c1cc(C)n(C)c1C)=O C12(CNC(c3c(C)nns3)=O)CCC1CCN2C(=O)CCCc1ncco1 N1(C(C(n2cnc(C#N)n2)C)=O)CCC(C)(NC(=O)CSc2ncccn2)C1 c1(C(N2C(C)CN(C(CCC=C)=O)C(C)C2)=O)coc2c(F)c(Cl)ccc12 c1(C(N(CC(=O)NCC(C)(O)C2CCC2)C2CC2)=O)ocnc1C(F)F c1(NC(c2c(Cl)cccc2Cl)c2n(CC)nnn2)cc(O)ccc1C c1(CCC(=O)NC(C2CC(NC(c3nccn3C)=O)C2)C)ccccc1N(C)C c1(C(N2CC3CC3C2)=O)cc(-c2ccccc2C(F)F)cc2[nH]ncc12 C1(C(=O)NCC(CN(C(c2c(C)cc(F)s2)=O)C)O)CC2(C1)CC21CCC1 C(=O)(CCCC(=O)N(C)CC1CCCC1NC(C1CCC(OC)C1)=O)OC Cc1ccc(C(C)NC(C2(C(C)NC(C3CCCN3C)=O)CC2)=O)nc1 C1(CNC(C2(C)ON=C(C)C2)=O)CC2(C1)CN(C(=O)CC1CN3CCC1CC3)C2 C1(NC(C(C2CCC(=O)N2)C)=O)(CNC(C2CNC(=O)N2)=O)CCCCCC1 C(=O)(C1CCc2cccnc21)NCC1CN(C(COCCC(C)C)=O)CC(C)C1 Cc1cc(=NC2CCCc3c(O)cccc32)[nH]c(N2CCC(c3ccn[nH]3)C2)n1 c1(NC(C(COCC)N=[N+]=[N-])=O)cccc2c1OCCO2 CON(C)CCCNC(=O)CC1CCN(C(=O)CC2(O)CCC2)C1 c1(C(C(=O)NCC2C(C)(C)OCC2)(F)F)cc(C(F)(F)F)cc(F)c1 C(=O)(C1=NN(C)C(=O)CC1)NC1CN(C(C(COCC)C)=O)CC2(C1)CC2 C1(NC(CCNC(=O)OC)=O)CCN(C(C2CC(OC)C2)=O)C1 S(=O)(=O)(c1cccc2c1OC(C)C2)N1CC(c2c(CC)nco2)C1 S(=O)(=O)(c1ccc(-c2sc(C(=O)OC)c(C)n2)c(OC)c1)NCCSC S(=O)(=O)(c1ccc(F)c(F)c1)N1CCC2(CC(C(N3C(CO)CC(C)C3)=O)C2)CC1 N1(C(C2CN(C(C(C)c3ccsc3)=O)CC2C)=O)CCC(O)CC(C)C1 c1(CN=C(NC(CC)CC)NC(CO)CCF)cn2ccccc2n1 C(=O)(C1c2ccccc2C(=O)N1C)N1CC2CC(CN(C(C(C)CN(C)C)=O)C2)C1 c1(C(=O)Nc2ccc(SC)c(F)c2)cc2n(n1)CCCN(C(=O)C(C)Br)C2 Cc1ccc(F)c(C(=O)NCC(C)(O)CNC(=O)CC2OCCO2)c1Br c1(C(=O)NC2(CC#C)CCC2)c[nH]nc1OCC N1(C(c2cc(Cl)cnc2O)=O)C2CCC1CC(NC(C1(O)CC3CC1C3)=O)C2 c1(C(=O)NC(CCCNC(C(C)NC(=O)C(C)(C)C)=O)C)cccc(F)c1C#N c1(N2CC(CN(C(c3cnc(CC)nc3O)=O)C)C2)nc2cc(C)ccc2s1 N1(C(C2(NC(=O)Cn3cccn3)CCN(C)C2)=O)CCN2CCOCC2C1 C(=O)(CC(C(=C)C)OCC)N1CCC(NC(CCOCC#C)=O)C1C N1(C(C(=O)NC(C)C)=O)CC(NC(=O)C(C)OCCN(C)C)C(C)C1 Cc1cn(CC(=O)NC2(CN(C)C(C3CC(F)(F)C3)=O)CC2)nc1C(F)(F)F C1(CC(=O)NC(CNC(CC(CCC)O)=O)C2CCC2)CCC2(CCCC2)CC1 C1(F)(C(N2CCC(CCNC(c3c(C)n[nH]c3)=O)CC2)=O)CCC(C)CC1 N1(C(C2N(C(C(C)=CCC)=O)CCC(CC)C2)=O)CC(C2=NOC(C)C2)C1 C12(NC(=O)CC3CC3)CCC(C1)N(C(=O)C(=O)NC1(C(F)(F)F)CCCC1)C2 c1(C(=O)NC(C(CO)NC(C(CC)SC)=O)C)cnn(CC)c1C1CC1 C1(NC(Cc2c(C)n(C)nc2)=O)CN(C(C2CC2(F)F)=O)CC12CC2 CC(C)C(O)C(C)C(=O)NCC1(C)CCN(C(C2CCN(C)CC2)=O)C1 c1(OC)cccc(C(N2CCC=C(CNC(C3(C)CSC3)=O)C2)=O)c1O c1(NC(C2CN(C(C3CCC(C(N)=O)C3)=O)C2)=O)ccc2nccn2c1 N(C(=NCCCCC1CCCC1)NC1CCCC1)Cc1cn(C)nc1C(F)F C1(C(=O)NCC(C2CC2)NC(C=Cc2n(C)ncc2)=O)CN2CCC1(C)CC2 c1(NC(C2C(NS(C(C)C)(=O)=O)C2)=O)cccc2c(Cl)ccnc12 CC1(C)CC(C(N2CCC(CO)(NC(c3occc3F)=O)C2)=O)CCO1 c1(C(=O)NC2CC2CNC(C2CCCCO2)=O)cccc(F)c1F C1(CNC(c2c(N(C)C)cncc2)=O)CC2CCC1N2C(c1scnc1Cl)=O c1(N2C(C(=O)NC(CC)C)CC(O)C2)ncnc2ncc(Br)cc12 N1(C(c2ccc([N+](=O)[O-])cc2OC)C(=O)NC)CCOC2(CCC(F)(F)CC2)C1 c1(CNC(COC)=O)ccc(N2CCN(C(C3CCCS3(=O)=O)=O)CC2)c(F)c1 [N-]=[N+]=NC1CCC(C(=O)NCCC2CC(F)(F)CN2C(C2CCNC2=O)=O)CC1 c1(C(=O)NCC2C3CN(C(COCCC)=O)C2C3)ccc([N+](=O)[O-])[nH]1 n1(CC)nc(C)cc1C(=O)NC(C(=O)N(C1CC(C)C1)C)C1CCC1 CC(O)CCCCCC(=O)NC1CN(C(c2ccc(CO)o2)=O)CC1C1CC1 CC(C)C(CN(C)C)C(=O)NC1CCC(NC(=O)CCc2cncc(O)c2)CC1 c1(C(=O)NC(C(C)C)C(C)NC(c2cnsn2)=O)cc(O)c(F)cc1N Cn1c(C(=O)NC2CCC(CNC(C3CC4CC3C3CC43)=O)C2)cc(Cl)c1Cl C(=O)(CC1OCc2cc(Cl)ccc21)NC(CC=C)CNC(C1CC2(CSC2)C1)=O O=C(C1=CCCOCC1)NCC12CCC(CN(C(=O)CCC(=O)NC3CC3)C1)C2 C1(CC(=O)NC(C=C)CO)CN(C(c2ncoc2CC)=O)CC1C c1(C(=O)NC2CCCN(C(C(C3CC3)OCC)=O)C2)ccc(CO)c(Cl)c1 c1(C(=O)NC2CC(C)(CNC(C3(C)CC=CCC3)=O)C2)csc2ccccc12 CC(C)C(C)(C(=O)N1CCC1CNC(=O)CCNC(N)=O)c1ccccc1 c1(NC(C2C3CCN(C(C(C=CC)O)=O)CC32)=O)ccc2c(c1)COC2 N1(C(c2c(OC)cnc(F)c2)=O)CCCC(NC(C2CCC(=O)N2C)=O)CC1C Cc1nc2c(s1)CCCC2C(=O)N1CCC(OCCNC(C2CC=CCC2)=O)C1 CC1(C)CC(NC(C2(n3ccnn3)CC2)=O)CC(C)(C)S1(=O)=O CC1(CNC(=O)C(F)=C2CCC2)CC(F)(F)CN1C(C1CCc2nnnn2C1)=O N1(C(C(CC)n2nccc2C)=O)CCc2nc(CNC(=O)COCCF)sc2C1 c1(C(N2CCCC(N(C(=O)C(F)=CC3CC3)CC)C2)=O)cncn(C)c1=O C1(NC(COC2(C)CN(C(C3C(C)(C(=O)OC)C3)=O)C2)=O)CCC(F)(F)CC1 C(=O)(C1CCc2cc(F)ccc21)N1CCC(C)C(CNC(C2CCCCO2)=O)C1 CCCC(C)CC(=O)NCCC1CN(C(c2cncc(O)c2)=O)CCO1 C1(C(=O)NCC2(CC)CCCC2)(CC)CCN(C(C2CCCC2)=O)C1 C(=O)(C1=CCCCCC1)NCCC(C)N(C)C(C1CCC2(CCC2)C1)=O N1(C(c2c(C)cc(C)o2)=O)CCCC(F)(C(=O)NCCc2ncccn2)C1 C#Cc1cnc(NC(C2CC2NCc2ccc(C(F)(F)F)c(F)c2)=O)cn1 N1(C(C(C2CCCOC2)OC)=O)CCCC(N=c2cc[nH]cc2[N+](=O)[O-])CC1 N1(S(c2c(C)nn(Cc3ccc(C)cc3)c2C)(=O)=O)CCC(C)CC1C1CCC(C)O1 c1(C(N2CCC(O)(CC)CC2)=O)cnn2c1CNCC2 C(C1(C)CCOCC1)=CC(=O)NC(CNC(c1c(C)sc(O)n1)=O)CO CC1CCN(C(c2cnc(Cl)[nH]2)=O)C(C)C1NC(c1cn(C2CCCC2)nn1)=O c1(CC(=O)NC(CCNC(C(CC=C)C)=O)C)c(F)c(F)cc(F)c1F Cc1cc(=NC2CCCN(C(=O)Cn3cc(C4CC4)nn3)C2)[nH]c(CO)n1 Cc1cc(=O)c(C(=O)NC2CC3CN(C(=O)Cn4nccc4N)CC23)cn1C C(CC(C(C)C)NC(=O)CCCc1csc(=N)[nH]1)NC(C1CC(SC)C1)=O N1(C(c2c(C)occ2)=O)CCCC(NC(=O)Cc2cccc(Br)c2)C(F)C1 C(=O)(CCC(=O)NN(C)C)NC(C)CCNC(C1CCSC1)=O N1(C(CCc2n(C)ccc2)=O)CC2CC(NC(C3CC(=O)NC3(C)C)=O)C1C2 CC1=C(C(=O)N2CCOC(C3CN(C(=O)CC(C)N(C)C)C3)C2)CC1 C(CC(C)C)(CS(=O)(=O)NC1CCN(S(C)(=O)=O)CC1C)OC Cc1cc(-c2cc(CN3CCOC(CO)C3)ncn2)c(F)cc1O c1(OC(C)C)cccc(C(=O)NCC2(F)CN(C(=O)CC3CN(C)CC3O)C2)c1 C(C)(CCC(=O)NCC1CCN(C)C1)NC(c1ccc(CC)[nH]1)=O CC(C)CC(F)C(=O)N1CC=CC1CNC(=O)CCCSC(C)(C)C C(=O)(CC(C)(C)O)N(C1CCN(C(C23CCCC2(C(N)=O)C3)=O)CC1)CC#C c1(COC)nn(C)cc1C(=O)NCC(C)(O)CNC(=O)CCSC1CCCC1 c1(OCC)cccc(CC(=O)NC2(CO)CCN(C(=O)CN(C3CCC3)C)C2)c1 Cc1nc(C)n(CCC(=O)NCCC(C)NC(=O)COC2CC=CC2)n1 C[Si](C)(C)CCCC(=O)N(CC(F)(F)F)Cc1cccs1 C(C(CC(=O)NCC(C1CCCCC1)O)OC)NC(c1ccn(CCC)n1)=O C(C(O)CC(=O)NCC1(C(=O)NCC2(C(=O)NC3CC3)CCN(C)C2)CC1)N(C)C c1(CCNC(=O)NC(c2ccco2)COC)cccc(SC(F)(F)F)c1 Cc1nn(C)c(C)c1C(=O)NC1C2CC1N(C(C1SCCS1)=O)C2 CN(CCCCc1ccc(F)cc1)N1CCC(C(N)=O)(CO)C1 C1(NC(CC2(COC)CC2)=O)CCN(C(=O)C(O)Cc2[nH]cnc2C)C1C N1(CC)N=C(C(=O)N(C)CCNC(c2nn[nH]c2C(F)(F)F)=O)CCC1=O N1(C(C2C(NC(c3c(C)oc(C#N)c3)=O)CCCC2)=O)CC2(CCC2)CC1C N1(C(CSCC)=O)CCCC2CN(C(c3ccc(C(F)(F)F)o3)=O)CCC12 c1(CC2(C(=O)OC)CCC2)ccc2c(c1)ncn2C.C12CC13CN(C3)NC2=O C=C1CC2(C1)CC(C(=O)OCc1sc(Cl)cc1Cl)C2 Cc1cnc2ccc(C(=O)NCCC3CN(C(c4cc(Br)n(C)c4)=O)C3)cn12 N1(C(C(C(C)C)SC)=O)CCC(C(=O)N(C2CCCN(C)C2)C)=C(F)C1 N1(C(C2(C(=O)NC)CCC2)=O)CCC(C)(CC(=O)NC2CC(C(C)(C)O)C2)C1 c1(NC(=O)OC(C)(C)C)cc(CNC2C=CCC2)cc(C(F)(F)F)c1 C1(COC(c2cccc(SCC)c2)=O)CCC2(CC(C(=O)O)C2)O1.C1CC1 Cn1cnc2cc(C#N)nc(N3CCN(C(c4ccc(F)cn4)=O)CC(O)C3)c12 C(=O)(C1=CCC1)NCCN(C(C1CC(C(C)(C)C)C1)=O)Cc1ccccc1 N1(C(=O)NCCc2cc(C(F)(F)F)ccc2Cl)CC2CC(F)(F)CC2C1 N1(C(C(C(C)C)N(C)C)=O)CCC12CN(C(C1CCCN1c1ccccc1)=O)C2 c1(CC)ccc(F)c(C(=O)NC2C3CCN(C(c4cnnc(O)c4)=O)C23)c1 c1(NCc2cc([N+](=O)[O-])c(O)cc2)cc(-c2cscn2)nc2ccccc12 C1(CNC(c2ncc(OC)cn2)=O)(NC(=O)CC(C)C(C)C)CCCCC1C CC(C)CCN=C(NCC1CC1)N1CCC(C(O)C(F)(F)F)CC1 C1(CNC(CSCCCC)=O)(NC(=O)Cc2ccc(C(F)F)cc2)CCOCC1 O=C(CC1COCc2ccccc21)NC1CCN(C(=O)Cc2ccns2)CC1O c1(C(=O)NC2C3CN(C(C(CCC)CCC)=O)CC32)cnc2cc(O)nn2c1N C1(CNC(C2CN3CCCN2CC3)=O)CCN(C(c2cscc2Cl)=O)CC1(F)F C1(NC(c2c(C)cc(C)nc2)=O)CN(C(=O)Cc2nc[nH]n2)C2CCCC12 c1(C(=O)NCCCNC(c2cnn(CC)n2)=O)ccc2c(c1)C(C)CO2 c1(N(C)C)c(C(=O)NCCCNC(=O)C(C)(C)C(N)=O)nnc2ccccc12 C(CC(O)C(=O)NC1(C(=O)NCC23CCC(CC2)C3)CC(F)(F)C1)N(C)C n1(CCC)nc(C)cc1C(=O)N(C(CNC(=O)C(C)O)CC)C C1(C(=O)NCCc2nc(C)on2)N(C(C2CC(C)C2)=O)CCCC1(C)C C1(CNC(Cn2cc(C(C)=O)nn2)=O)CCCCN(C(c2cncnc2)=O)C1 CC#CCC(C(=O)NCC12CCCC1CCO2)NC(=O)C=CCN1CCC1 C1(OC)CCC(C(=O)NC(C2CC=CCC2)C(=O)NCCN2CCOC2=O)CC1 C1(O)(C(COC(C(=O)OC)OCC)C)CCN(C(=O)CCc2csnn2)C1 n1(CC)nc(C(N2CCC(Cc3cccc(F)c3)C2)C(=O)NCC(C)C)c(C)n1 C1(CC(=O)NCc2nccs2)CCCN(C(=O)CC2CCCCO2)C1 C1(C(N2CCC(C(=O)OCC)C2)=O)(NC(C(C)OCCCC)=O)CC1(C)C c1(C(=O)NCC(CC)NC(=O)Cc2csc(C)n2)c(C)oc(C)c1C CCC(CNC(=O)Nc1cccc(CN2CCCC2=O)c1)(CC)SC N1(C(C2(COC)CC(=C)C2)=O)CCCC2(CCN(C(C3SCCCS3)=O)C2)C1 c1(COCC(=O)NC2CCC2NC(c2cocc2Br)=O)cccnc1 C(=O)(C(C)(C)S(C)(=O)=O)NC(CC)CNC(C1CCCCC1(F)F)=O Cc1ncc(CC(=O)NC(C)C(CO)NC(c2cnc(N(C)C)s2)=O)s1 c1(CNC(c2ccc(F)cc2)C(C)(C)O)nc2cc3c(cc2[nH]1)OCO3 N1(C(c2n(CCC#N)ncc2)=O)CCC(CNC(C2(n3cccn3)CC2)=O)CC1 c1(OCC)c[nH]nc1C(=O)NCCCCCOCCNC(=O)Cc1ccco1 n1(C(C)C)cnc2c(N3CC4CCC4C3)[nH]c(=NCC3CCC(C)(C)CC3)nc12 C(c1ccccc1C#N)=CC(=O)NCC1(C)CCCN(C(CC2(C)CCC2)=O)C1 N1(C(c2c(C)cnnc2)=O)C2CCCC1CN(C(c1coc3ccccc13)=O)C2 N1(C(C2CCN(C(C(CC)O)=O)CC2)=O)CCc2c(C#N)cccc21 C1(N(C(=O)CCn2cc(Cl)cn2)CC)CCCN(C(=O)CC2(O)CCOC2)C1 C(CCCCCC(=O)NC1(C)CCC1)n1cc(C(CCC)NCCOCC)nn1 C1(NC(C2CCCN(CC)C2)=O)CCN(C(=O)CC2CCCC2)CC1(C)C C1(O)(C(C)NC(c2nocc2Br)=O)CCN(C(C2COCCOC2)=O)C1 Oc1ccc(CNC2CC3(C2)CC3(F)F)cc1OCC(F)(F)F C1(CNC(Cc2c(C)ccnc2)=O)CCN(C(C2CCCNS2(=O)=O)=O)C1(C)C Cc1cc(=NCc2cccc(O)n2)[nH]c(=NCC2CCCOCC2)[nH]1 C1(NC(c2ccc(O)nn2)=O)CN(C(=O)C#CC2CCCCO2)CCC12CCC2 c1(NC(C(C)N(C(C(CC=CCC)C)=O)C2CC2)=O)ccc(F)c(O)c1 c1(OC(C)C(=O)NC(c2nnc(-c3ccccc3F)s2)C)cc(Cl)ccc1CO c1(SC)cccc(C(=O)NC2CCCCC2NC(=O)Cc2cnnn2C)c1Cl C1(C(N(C(=O)CCNC(=O)CCN(C)C(=O)OC)CC)C)CCC1CO c1(SCC(=O)NC23CC(CNC(C4CC(F)(F)C4)=O)(C2)C3)ccncc1 c1(C(=O)NCC2C(NC(C(COC)OC)=O)COC2)cccc(CS(C)(=O)=O)c1 c1(C(F)F)nc(-c2ccc(I)cc2)n(CC2CCC2)n1 C1(CCNC(COC)=O)CCN(C(c2cc(OC)cs2)=O)C(C)C1 C12(C(=O)NC3C(CNC(Cn4c(C)ncc4)=O)CCC3)CCC(C1)OC2 c1(C(=O)NCC2(F)CC(CNC(C(c3ccccc3)SC)=O)C2)ccn(C)c1C c1(C2CCN(c3n(CCC)c(C4CCOC4)nn3)CC2)nc2c(s1)CCC2 c1(C(C)OCC)nc(C)c(C(=O)N(CCCNC(C2CCOC2C)=O)C)s1 c1(C(=O)NC2CC(CCNC(C3(F)CC3)=O)C2)nc2n(c1Cl)CCCC2 N1(C(c2ccc(OC)cn2)=O)CCN(C(C2(C)CCCCC2)=O)CC1CCO C1(C(=O)NC2(C)CCN(C(C(C)=C(CC)C)=O)CC2)CCN(S(=O)(=O)N(C)C)C1 N1(C(C(Cc2c(C)n[nH]c2C)C)=O)CCC(C)(NC(=O)CC2CC23CC3)CC1 C1(CNC(C(COC)C)=O)CCCCC1NC(c1ccn(CC2CC2)c1C)=O C12(NC(C(C)OC)=O)CCOCC1CN(C(c1ccc(Br)cc1F)=O)C2 C1(NC(C=CC(C)(C)C)=O)CC2CCC1N(c1cc(-n3ccnc3)ncn1)C2 c1(C(=O)NCCC(C)N(C)C)cc(Cl)ccc1NC(=O)CN1CCCCCC1 c1(C(=O)NCCCN(C(C2CCCCC2(C)C)=O)CC)nccc2ccccc12 c1(C2N(CC(COc3ccc(OCC)cc3)O)CCC2)ncc(F)cc1F C1(CC(N)=O)CCCN(C(=O)C(Cn2cccn2)NC(C2CCOCC2)=O)C1 c1(C(N2C(C(=O)NCc3cc(C)c(F)cc3)CC(O)C2)=O)ccc2ncnn2c1 c1(OCC(=O)NCC(CC)NC(C2COC(=O)N2C)=O)ccc(C)cc1C C(=O)(C1=Cc2cc(F)ccc2OC1)NCC1CCN(C(CC(C)O)=O)C12CC2 C1(C(C)C)CN(C(C2C3CCN2CC3)=O)CCN1C(c1cc(C(F)F)[nH]n1)=O C1(CC)COC(C)CN1C(c1scnc1C)C(=O)Nc1ccccc1 N1(C(C(N2CCC(NC(CC3ON=C(CC)C3)=O)CC2)=O)C)CCP(C)(=O)CC1 C1(CNC(c2cn(CC)nc2)=O)CCC(C)CN1C(c1cc(C(F)F)ccn1)=O C1(C(=O)NC(CNC(c2ccc(C#N)o2)=O)CO)CCC2(CCC2)OC1 c1(OC)cccc2cc(C(=O)NCCNC(=O)CC(C)SCC(C)O)c(=O)oc12 C#CCC(CC)NC(=O)C(CSCC)NC(=O)C(C1CCC1)OCC c1(N(C(c2c(C)ccc(C)c2N)=O)C)ccc(S(=O)(=O)C(F)(F)F)cc1 C1(CN(C(=O)CCCc2ccccc2)C)CCCN(C(C2(CF)CC2(F)F)=O)C1 c1(C(=O)NC2CN(C(Cc3c(C)con3)=O)C(C)C2)ccccc1P(C)(C)=O N1(C(=O)CCSc2ccc(Br)cc2)CC2(CCCC2)C1C(=O)O N1(C(CC2(C=C)CCC2)=O)CC(CNC(c2cn(CC)nn2)=O)C2(CC2)C1 c1(C(N(C2CCN(C(c3ccc(Br)c(F)c3F)=O)C2)C)=O)ccc([N+](=O)[O-])cc1 Cc1ccn(C(C)C(=O)NC(CO)C(=O)NCC2(CO)CC=CC2)n1 C(=O)(CC(C)(C)C(F)F)NC(C(C)C)CCN(C)C(C1CC(C)(C)C1)=O c1(C(=O)NC2(CCOC)CCN(C(C3CCC3C)=O)C2)cncn(C)c1=O C1(CC)(CC)CC(NC(c2c(C)nn(C)c2C)=O)CN1C(=O)Cc1nccn1C CCCCC(C(=O)Nc1ccc(C(C)C)nc1)NC(=O)C(CC)C(C)C c1(OCC)cc(Br)ccc1NC(C1CCC(NC(=O)C=Cc2cnccn2)C1)=O N1(C(c2cccc(CC)n2)=O)CCCN(C(=O)C(C)OCC2CC2)C(C(C)C)C1 c1(NC(C2N(c3ncc(C(=O)OC)cn3)C3C(C2)C3)=O)ccc(Br)cc1O N1(C(CCNC(=O)Oc2ccco2)=O)CC(F)(F)CC1CNC(C1CCCO1)=O C12(C(=O)NC3CC(N(C)C(c4ncn5c4CCC5)=O)C3)CCC(C)(CC1)CO2 CCS(=O)(=O)c1ccc(Cl)cc1C(=O)NCC1CN(C)CCN1C(C1CC1F)=O c1(C(N(C(CCC)C)C)=O)cncc(CNC(=O)CCC2CCC(C)O2)c1 CCCS(=O)(=O)C(C)C(=O)NCCN(C(=O)C(C)=C1CCCC1)CC1CC1 c1(CNC(=O)CCCOc2ccc([N+](=O)[O-])cc2)c(F)ccc2[nH]cnc12 C(=O)(C(CC(C)CC)NC(=O)C(C)CCN(C)C)N1CC(CC)N(C)CC1 CC1CCCC=C1C(=O)NC(C)C(CO)NC(=O)Cc1ccc(F)cc1Br Cc1cc(N)cnc1C(=O)N(C1CCN(C(C2CCC3C2C3(F)F)=O)CC1)C N1(C(CN(c2nnc(S)n2C)C)=O)CC(C)(C)C1C1CCCO1 Cc1cc(C(=O)NCC2(CNC(=O)C(F)C3CCCC3)CC2)c(C)n1C Cc1ccc(C(=O)NCC2C3CCC(C3)N2C(c2n[nH]c(C)n2)=O)c(C)n1 S(=O)(=O)(c1cnc(C2CC2)nc1)NCC1OCC(C)C1 C1(F)(C(=O)NCC(CNC(c2cccc(Cn3cccn3)c2)=O)O)CCCOC1 c1(C(=O)NC2COCCN(C(C(C3CC3)OCC)=O)C2)ccc2c(n1)CCO2 CC(=NO)C1CC(C(=O)N(CC(C)NC(=O)C=Cc2ccccn2)C)C1(C)C c1(C(=O)NCC23CCC2CCN3C(c2ncccn2)=O)cc2c(cn1)OCCO2 N1(C(C(C=C)O)=O)CC(C)OC2(CCN(c3ccc([N+](=O)[O-])cc3C(F)F)C2)C1 C(CCC(N)=O)(C(=O)OCC1CCNC1=O)N(C)C(=O)OC(C)(C)C C1(CNC(N2CC(C(=O)NCC(F)(F)F)C(C(F)(F)F)C2)=O)CC2(CCC2O)C1 C(=O)(C1=CCC(C)CC1)N(C1CCCN(C(=O)CN2CCOCC2)C1)CC N1(C(C(=O)NCc2c(C(C)(C)C)cccn2)=O)CCc2ccccc21 N1(C(Cc2nc(C)[nH]n2)=O)CC(NC(c2ccc(N)c(O)c2)=O)CC12CCCC2 c1(C(=O)NCC(C)NC(c2ccc3cn(C)nc3c2)=O)cnn2c1CC(C)CC2 c1(CC)noc(CNC(=O)C(=O)N(C2CCCC2C)CC)n1 C1(C(=O)NCC(CNC(=O)C#CC2CC2)C(F)(F)F)(NC(C)=O)CCC(C)CC1 N1(C(C(C)Cc2ccncc2)=O)CCC(NC(=O)CCN2CCCC2)C(C)(C)C1 N1(C(C)C)CC(C(N2CC(NC(=O)CC3CC3)C(c3cncn3C)C2)=O)CC1=O C1(C(N2CCCC(O)C2)=O)CC2CCC(C1)N2C(c1ccn(C(F)F)n1)=O C1(OCC)COCCC1CC(=O)Nc1cccc(NC(=O)Cc2ccsc2)c1 C1(CNC(C2(C#N)CC2)=O)CN(C(C2CCN2C2CCCC2)=O)C2(CCC2)C1 CCN=c1ccc(C(=O)NCC2C3CN(C(=O)CCS(C)=O)CC23)c[nH]1 C1(NC(COCCCOC)=O)CCC(NC(=O)CN2CCCC2CO)CC1 Cc1[nH]nc(Cl)c1C(c1nnnn1CCN1CCOCC1)NCC1(C)CC=CCC1 N1(C(c2cc(C)oc2)=O)CCCC2(CC(NC(=O)C(C)(Cl)Cl)CO2)C1 N1(C(c2n(CC)ncn2)=O)CCC(NC(c2ccc(Cl)cc2C)=O)C(F)(F)CC1 O=C(CC(C(F)(F)F)n1cccn1)NC1CN(C(=O)C(F)(F)CN2CCCC2)C1 N1(C(Cc2ccn(C)n2)=O)CCC2(CCCCC2NC(C2CC2F)=O)C1 c1(CSC)cccnc1C(=O)NC(C)CCN(C)C(c1ncccc1N)=O CC(=O)C(C)CC(C)C(=O)NC1CCC1NC(C12CC(F)(C1)C2)=O CCCCC(CC)C(=O)Nc1ccc(C)cc1.c1(C2CCN2)cccc(Cl)c1.OC c1(OCC)ccc(S(=O)(=O)N2CC(C)(CO)C2)cn1.c1(C=O)cncn1C C1(N(C(C=C(CC)C)=O)C)CCCC(N(C)C(C2CCC(C)CC2)=O)C1 c1(N2CC(COC)N(C(C3CCCCCC3)=O)CC2)ncc2ccccc2n1 Cc1cc(-n2cccn2)nc(NC2CCN(C(=O)CCCC3CCC3)CC2C)n1 C(=O)(C1=NOC(C)C1)Nc1cc(C(=O)NCc2ccccc2)on1.C12CC1C2N N1(C(C(C)OCc2ccc(F)cc2)=O)CCN(C(=O)CC23CC(C2)C3)CC1C c1(SCC(=O)NC(c2cnn(C3CCCCO3)c2)=O)cccc(F)c1 c1(CC(=O)NC23CC2CN(C(=O)Cn2cnnc2)C3)coc2ccccc12 c1(N2CC(CCC)OCC2)nc2cccc(F)c2c(=NCc2ccoc2)[nH]1 N1(C(C(=O)NCC2(C(F)(F)F)CCCC2)=O)CCOC2CCCCC12 c1(C(=O)NCc2c(C(=O)NC(CCC)C3CC3)scc2)ccccc1OCC N1(C(C(C=C=C)C)=O)C2CCC1C(C(=O)NC(CF)C(F)(F)F)C2 Cc1ccnc(C(N2CCC(N(C)C(c3ncc(F)cc3F)=O)C(C)C2)=O)c1F C1(c2nnnn2CCCOC)(NC(CCC)CCOC)CN(C)CC1C C1(NC(c2c(CC)c[nH]n2)=O)CC2CCC1CN2C(=O)C(c1ccccc1)C CS(=O)(=O)C1CN(C(=O)Cn2ncnn2)CC1NC(C1(CC(F)F)CC1)=O c1(CN2CC(NC(c3cc(C)cc(Cl)c3)=O)C2)cc([N+](=O)[O-])cc(Br)c1O Cc1cccc(F)c1C(=O)NC1(C(N2CCCC(CC(N)=O)C2)=O)CC1C C(N1CCC(F)C1)N1C(=O)CCC1 c1(C(=O)NCC2(C#N)CN(C(c3ccc(C)n3C)=O)C2)cc2ccccc2[nH]1 C(=O)(C(C(C)(C)C)n1ccnn1)N1CC(C(C)NC(c2csc(O)n2)=O)OCC1 Fc1cccc(C2CCCCN2c2cc(Br)ncn2)c1 c1(CNC(CCOC(C)C)=O)cc2cc(F)ccc2[nH]1 C(C(CO)CC(C)C)NC(CN(CC(C)C)C(=O)CC1CCCC(=O)C1)=O N1(C(c2cc(C)oc2)=O)CCC2CCCC12CNC(c1cnn(C)c1N)=O N1(C(CC2(C(=O)OC)CC2)=O)CCC2CN(C(c3ccc(CO)cc3)=O)CCC12 c1(C(N(CCN(C(CC2C(CC)C2)=O)C)C)=O)cc(S(=O)(=O)N2CCC2)c[nH]1 CCC(C)C(O)C(=O)NCC(C1CCC1)NC(c1cnn(C)c1SC)=O c1(OCC(=O)NCCCN(CCCNC(C(F)OC)=O)C)cc(Cl)ccc1Cl Cc1cccc2c(O)nc(-c3ccc(N4Cc5ccc(O)cc5C(C)C4)cc3)nc12 c1(OCC)c(Br)cc(CN(C)Cc2ncc(C)n2C)cc1Br S(=O)(=O)(c1ccc(C(=O)OCc2cc(C)ccc2C)cc1)NCC N1(CC(N2CCC(C(N3CCCCC3CCCO)=O)CC2)=O)CCC(O)CC1 c1(OC(C)C)ccc(C(N2CCN(C(C3CCN(C)CC3)=O)CC2C)=O)c(F)c1 N1(C(CNC(=O)CC2CCCC2(F)F)=O)CCN(C(c2coc(O)n2)=O)CC1 N1(C(C(=O)NC(C2CC(O)C2)(C)C)=O)CC(C(F)F)C2(CCC2)C1 CC1CN(C(=O)C#CCNC(=O)C(F)CC2CCOC2)CCN1C N1(c2nnc(C(C)OC)n2CCc2ccc(Cl)cc2)CCS(=O)C(C)C1 c1(CC(=O)NC2CCCC(NC(C(C)OC)=O)C2)cccc([N+](=O)[O-])c1C C1(C(=O)NC(C2(O)CCN(C(c3cnn(C)c3)=O)C2)C)CCCCCCC1 c1(C(=O)NC2(CNC(CNS(CC)(=O)=O)=O)CCCC2)cc2ccc(F)cc2[nH]1 C(=O)(CCCCC(C)(C)C)N1CCC(NC(C(CC=C)C(C)C)=O)C12CC2 O=C1CC2(CCC2)C(C(=O)NCCCCNC(=O)C2=CCCO2)CN1 C1(NC(=O)Cc2cccc(Br)c2)CC2C1CCN2C(=O)CSc1ccon1 CCC(F)(F)C(C)(C)C(=O)N(CCC(C(C)C)NC(=O)CCC(C)C)C CC(C)CC(C)NC(=O)C(C)NC(=O)CNC(C1CCCC1)=O c1(COCC)ccc(CN(c2ncc(-c3ccccn3)s2)C=O)s1 c1(CNC2CC(OC(C)(C)C)C23CCC3)ccc2c(c1)N(C)CC2 C1(C(=O)NC2CN(C(c3c(C)scn3)=O)C(C)C2)CC12CCSCC2 c1(CNC2CC(NC(C3C(C)C3)=O)C2)ccc(Cl)c([N+](=O)[O-])c1 CC(O)CCN=c1cccc(S(=O)(=O)NCCc2ccncc2)[nH]1 C1(C(=O)NCC2C(NC(C(CC)CC3CCCCC3)=O)C2)CN(CP(C)(C)=O)C1 Cc1c(C(N2CC3C(CNC(c4cnc(O)o4)=O)C3C2)=O)oc2ccc(F)cc12 C(C(CNC(=O)CC1CCC(C)CO1)S(C)(=O)=O)NC(CCOCCOCC)=O Cc1c(C(N2CCC(NC(=O)C(C)(C)N3CCCC3)C2)=O)[nH]c2c(C)cccc12 C=CC(C)(CC)C(=O)NC(C)CC(C)NC(c1nc(Cl)ccc1Cl)=O CC1Cc2ccc(F)cc2C1NC(=O)CCCOCCCN c1(OC)cc(C(N2CCC(NC(=O)C3=CCC3)C(C(C)C)C2)=O)ccc1Cl c1(OCCC(=O)NC2CCC(NC(CC#N)=O)C2)ccccc1F c1(C(N2CC(CC(C)NC(=O)COc3ccc(Cl)cc3)C2)=O)c[nH]c(=O)cn1 C1(NC(C(C)C)=O)CCCC(NC(c2ccccc2-n2ccnn2)=O)C1 C1(C(=O)NC2C3N(C(c4scc(C)c4Cl)=O)C(CC3)C2)CCC2(CCOCC2)O1 C(=O)(C1=NOC(C2(O)COC2)C1)N1CC2C(N(C(=O)CC3CC4CC4C3)C)C2C1 N1(C(c2c(C)coc2C)=O)CC2=C(C1)CN(C(=O)C(C)Cc1cnc[nH]1)C2 c1(C(N2CC=CC2COCC2CCCCO2)=O)cc2n(n1)CCCN2 C1(NC(C2(C#C)CCCC2)=O)CC12CCN(C(c1coc(C#N)c1)=O)CC2 CC(CC(=O)NCC1C=CCN1C(C1(NC(=O)OC(C)(C)C)CCC1)=O)C(C)(C)C C12(CNC(c3c(CC)n(CC)nc3)=O)CC(CO1)N(C(=O)C(CO)N(C)C)C2 CC(c1cccc(Cl)c1)=CC(N1CC=CC(NC(C23CC2C3)=O)C1)=O n1(CC(N2C(CC)C(NC(=O)CN3CCCS3(=O)=O)CC2)=O)cnc([N+](=O)[O-])n1 N1(C(c2cccc(C(=O)NC)c2)=O)CC(C)CN(C(c2ncoc2C)=O)CC1C n1(CCC(N2CCC(c3cnccn3)C2)=O)cc(C2(F)COC2)nn1 CC1=C(C(=O)N2CC(CNC(c3oc(C)cc3C)=O)C3(CC3)C2)CCO1 c1(C(=O)Nc2nccc(C(N(CCC)CCC)=O)n2)ccc2csnc2c1 c1(C(N(C(C)CNC(=O)CCNC(=O)C2CC2)C)=O)csc(-c2ccco2)n1 N1(C(C(=O)NCC(=C)C)C2CCC2C(F)(F)F)CCN(Cc2cnc(Cl)s2)CC1 c1(OC)ccccc1C(=O)N(CCCCCCNC(C1CC(C)(C)O1)=O)C N1(C(c2cc(C(C)C)on2)=O)CCCC(O)C1C.C1C(=O)N1C(C)C C=CC1CN(C(c2c[nH]c(=NCC)s2)=O)CC1NC(=O)C(c1c(C)n[nH]c1C)C c1(C(N2CC(CNC(C(C)=C(C)C)=O)C(C)CC2)=O)cc(Cl)c2n[nH]cc2c1 N1(C(COc2cn(C)nc2)=O)CC2CCC1C1CN(C(=O)CCC(N)=O)CC21 c1(SCC(C)OC(C2CCCCC2C)=O)ccccc1Br c1(C(=O)NC2CCN(C(=O)CC3=CCCC3)CC2)cc2cccnc2o1 Cc1sc(N)c(C(N2CCC(C)(CNC(c3ccc(O)nc3Cl)=O)C2)=O)c1C C(CNC(C1(C)CC(NC(c2cc(CCO)on2)=O)C1)=O)(C(F)(F)F)OC C1(CCNC(C2CSC2)=O)CSCCN1C(=O)C=C1CCCC1 C(=O)(CC(C)(C(F)F)N(C)C)NC1(CO)CN(C(c2c(C)c(Cl)ccc2)=O)C1 C(=O)(C(C)(NC(C)=O)COCCCC(=O)NC1C=CC(CC(=O)C2CC2)C1)OC C(CC(C)(C)C)(C(=O)NCC1(F)CN(C(c2sc(C)nc2C)=O)C1)OC c1(CCC)onc(C)c1C(=O)N(CCC(=O)NC(c1ccccc1O)C)C(C)C N1(C(c2nc(C)c(C#N)cc2)=O)CCC2(CCN(C(c3cnc(Cl)[nH]3)=O)CC2)C1 c1(C(N)=O)cccc(CN2CCC(C(=O)NCc3ccncc3F)C2)c1 C1(NC(C(C=C)(C)C)=O)CN(Cc2nnc(Br)s2)CCC1C(F)(F)F C1(CN(C(C2CN(C(C)C)C2)=O)C)C2CN(C(C3(C)CC3(F)F)=O)CC12 C(=O)(CS(=O)(=O)C1CC1)N(C1CCCN(c2ccc([N+](=O)[O-])cn2)CC1)C C1(C)(NC(C(C)OCCC=C)=O)CCN(C(c2sccc2SC(F)F)=O)CC1 c1(C(N2C(C)CN(C(C3(CO)COC3)=O)CCC2)=O)ccc(N=S(C)(C)=O)s1 c1(OC)cc(C(F)(F)F)ccc1C(=O)NC1CCCCC1NC(=O)C(O)C(C)C C1(CC)(NC(=O)C(CN(C)C)N(C)C)CCN(C(=O)C=CC2CCCCC2)CC1 c1(C(=O)NCC2CCC(NC(CC3N(CC)C(=O)CC3)=O)C2)ccc(Cl)cc1F Cc1cc(C(N2CCN(C(=O)CCC(C)(C)C)CC2)=O)nc2ccccc12 C1(CNC(C(CCCC)F)=O)CCC2CN(C(C3(C#N)CCOC3)=O)CC12 N1(C(c2cnc(CC)[nH]2)=O)CC(NC(C2(C#N)CCCOC2)=O)CC12CCCC2 S(=O)(=O)(c1cnn2ccc(N3CCC(C)(N(C)C)C3)nc12)N1C(C)CC(C)CC1C N1(CC)CCCC(ONC(=O)C2(NC(=O)OC(C)(C)C)CC2C)C1 c1(CC)nc2c(C(=O)NCCN(C(=O)C(C)C(O)CC)C(C)C)ccnc2[nH]1 C1(N(C(c2ccc(CSCCC)o2)=O)C)CCN(C(=O)CC2(C)OCCO2)CC1 c1(OC)sc(C(=O)NCC(O)CN(C(=O)CC(C)OC)C)cc1Br c1(C(C(=O)NCCNC(c2cnn(C)c2)=O)N(CC)CC)ccc(SC)cc1Cl Cc1ccc2c(c1)C(N)C(C(N1CCC(Oc3ccc(C(N)=O)cc3)C1)=O)C2 N1(C(c2c(Cl)cc(C)nc2)=O)CC(NC(c2occc2C)=O)C(S(C)(=O)=O)C1 c1(C(=O)NC(CNC(c2cnn3ccsc23)=O)CO)c(Cl)ccc(F)c1F c1(-c2cn(C)nc2)ncccc1NC(=O)C(C1CC(F)(F)C1)O c1(C(=O)NCC2(C)CCN(C(C3CN(C)C(=O)C3)=O)C2)cncn(C)c1=O C(C)(CO)(C(=O)NCCCOCC1CC1)NC(C1ON=C(C)C1)=O N1(C(C=CSC)=O)CCN(C2COCC2NC(c2sccc2C(C)C)=O)CC1 N1(C(C=CC)=O)CC(CNC(=O)C(=O)NCC(F)F)C2(CCC2)C1 C1(CC(=O)NC(CSCC)C(=O)NCC2(C)CCN(C)C2)CCCN(C)C1 C1(OC)CN(C(=O)CN2CCCCC2=O)CC1NC(=O)C(C)CN(C)C N(C(=NCc1cccnn1)N1CCC2(O)CCOCC2C1)C(CC)C N1(C(C=C(CC)CC)=O)CCN(C(c2occc(=O)c2OC)=O)C(CCO)C1 c1(-c2onc(C3C(C)(CC)C3)n2)ccc(C(F)(F)F)cc1Cl CC1CN(C(c2ccon2)=O)CCC1N(C(=O)Cc1c[nH]ccc1=O)C C1(C)(CCNC(C=C2CCN(C)C2)=O)CCN(C(=O)CCc2ccc(O)cc2)C1 N1(C(C2(C)CC(C)C2)=O)CCC(C(C)C(=O)NCC2CCCOC2)CC1 C1(NC(COC)=O)CN(C(=O)C(C)Cc2ccc(Cl)cc2)CC12CCC2 C1(OCC(=O)NCCCN(C(=O)C(C)(C)F)CC)CCOCC1 Cc1cc(S(=O)(=O)N2CC3(CCCN3)C2)cc(C(=O)O)c1C c1(C(=O)NCC23C(CN(C(c4nc(C)sc4)=O)C2)C3)c(O)nnc2c1CCC2 Cc1cc(C(=O)NCCC2CC(NC(c3[nH]c(C)nc3C)=O)C2)c(O)nn1 N1(C(CCCOC)=O)CCC2(CCCN(CC3CCCO3)C2)C1.C1(=O)C(C)O1.OC C(=O)(CCCc1ccccc1)N(CCCCNC(C(C1CCCO1)OC)=O)C C(=O)(C(C(=O)NCCOCCCNC(c1ccoc1C)=O)OC)OCC c1(OCC)ncc(C(=O)NC2CCCC(C(=O)NCCSC)C2)cn1 c1(CC(=O)NCC(=O)NCC(C)NC(c2cccc(F)c2)=O)cccc(Br)c1 CC#CC1CCN(C(c2[nH]ccc2CNC(=O)C(C)C2CCCC2)=O)CC1 c1(N2CCC(C(C)(C)C)(CNC(C(CC)F)=O)C2)cc(C)nc2[nH]nc(C)c12 c1(CC)nc(C(N2CCC(NC(C3CN(CC)CCO3)=O)CC2)=O)c(N)s1 c1(CCC(=O)NC(C(C)C)CNC(=O)C(C)c2ncco2)ccc(C#N)cc1F c1(CC(=O)NCC(=O)OCCC2CC23CC3)cccc(O)c1 CN1CCOCC1C(=O)NCC1CC(C(F)(F)F)CN1C(=O)CCCC#N N1(C(c2cc(C)sc2N)=O)CCC2CCN(C(C3CN(C)CCO3)=O)CC12 C1(C)(C(C)C)CCN1C(c1ccc(CNC(c2coc(CO)c2)=O)s1)=O c1(C(=O)NC2CCCN(C(c3n[nH]c(C)c3C)=O)CC2)nnn2c1CCCCC2 c1(C(N2CCN(Cc3cc(Br)ncc3F)C3CC23)=O)ccc(Cl)c(Cl)c1 N1(C(C(C2CC2)OCC)=O)CCN(CC2CCN(C(C3CSC3)=O)C2)CC1 C12(CCCC1)C(=O)NC2.C(=O)(CN(C)C(C)=O)NC(C)C N1(C(C(C)NS(CC)(=O)=O)=O)CCN(C(c2cnc(O)cc2OC)=O)CC1C N1(C(c2c(CNC(c3ccc(CC)cc3)=O)ocn2)=O)CCOC(C)C1C CCC(C#N)(CC)C(=O)N1CC(N(C(=O)C=CCO)C)C2(CC2)C1 Cc1ccnc(O)c1C(N1CCC(O)C(NC(=O)CCOC2CCCC2)C1)=O CC(C)(C)CC(C(=O)N1CCCC1CF)NC(c1ccsc1)=O N1(C(C(N2CCC(CN(C)C(=O)OC(C)(C)C)CC2)=O)=O)CCc2ccccc2C1 N1(C(C(CNC(C(C(C)C)SCC)=O)O)=O)CC2(CC(O)C2)C1 c1(C(C(=O)NCCCC2CC2)N(CC)CC2(C)CCCO2)cc(Br)c(Cl)s1 c1(C(=O)NCCCCc2cnc[nH]2)cc(CNC(c2cnsc2)=O)ccn1 C(=O)(CC(C)(C)C(C)(F)F)NC(C)CCNC(C1(c2ccccc2)CCOC1)=O CCC(O)C(=O)OC.C1(CCOC(C)(C)C)CN1.C(=O)(C1CC1)O c1(-c2nc(CC(CC)C)nn2CCS(C)(=O)=O)ccnc2ccsc12 c1(C(C)OC)nc(C(=O)NC(C)(C)CCNC(=O)C(C)CC2CC2)cs1 c1(C(=O)NC2C(NC(CCCn3ncc(C)c3)=O)CCC2)cnn2ccn(C)c12 c1(OC)nn(C)cc1CNC(=O)C(=O)NCC(c1ccncc1)C C(CC(=O)NCCn1cc(CSC)nn1)(NC(COCC)=O)CN(C)C C=CCC(CNC(c1cnnn1C)=O)C(=O)N1CCC(N2CC=CC2)C1 C1(NC(c2ccc(C(C)(C)OCC)cc2)=O)C2CC1N(C(=O)C(C)C1CC1)C2C N1(C(CN(C(C)=O)C)=O)CCOCC(C)(CNC(C2CN3CCC2CC3)=O)C1 C1(C(N(CC(=O)NCC)CC)=O)CC2(CCN1C(=O)CSCC(N)=O)CC2 CC(C)C(N=[N+]=[N-])C(=O)NCCN1CCC(NC(C2CC2CCN(C)C)=O)C1 C1(CN(C(=O)C(c2ccccc2)NC(C2CC2(Cl)Cl)=O)C)CCCC1(C)C C(=O)(CCS(N)(=O)=O)NCC1C(CNC(CCOc2ccc(OC)cc2)=O)C1 C1(C)(C(=O)OC)CCN1C(C1(CNC(=O)C(n2cc(C)cn2)C)CCC1)=O NC1(CC(=O)NC2CC(=O)N(Cc3ccc(F)cc3F)C2)CCCS(=O)(=O)C1 C=CCCCC(C(=O)N(C)Cc1cncnc1)NC(=O)C(C1(C)CCOCC1)C C(=O)CCCC(C)(C)C.C(=O)(CCC(C)(C)F)N(C1CCN(C)CC1)C N1(C(COCC)=O)CC(CC(=O)N(C)Cc2ccncn2)CC1C C=CCN=C(NCCN(S(=O)(=O)c1cccs1)C1CC1)N1CC(C)N(C)C(C)C1 c1(C(C)C)ccc2cc(C(=O)NCCCN(C)C(C3CCS(=O)CC3)=O)[nH]c2c1 C(=O)(CC(F)(F)C(C)C)NCC1CC(NC(C(C)(C2CC2)OC)=O)C1 C1(C(=O)NCc2c(C)ccs2)CCN(C(c2c(C)nsc2C)=O)C(C)(C)C1 c1(OC(C(=O)NCCN(C(C2(OC)CC2)=O)C)C)ccccc1C C1(NC(c2ncccc2C(F)(F)F)=O)CC2CCC(C1)N2C(c1cc(O)no1)=O c1(NC(C(c2cc(Br)c(Cl)s2)N(C(C(CC)C)C)C)=O)cccc(OC(F)F)c1 c1(CC(=O)NCc2c(CCNC(C)=O)ocn2)cccc2cnccc12 c1(N(CCCNC(C)=O)C)cc(S(=O)(=O)NCC(O)C2CCC2)ccc1C#N C1(N(C(CNC=O)=O)C2CC2)(CF)CCN(C(=O)C(Cl)Cl)C1 N1(C(c2cc(CNC(C(CC#C)C3CC3)=O)on2)=O)C2CCC1CC(F)C2 C(=O)(C(CC)CCOC)NC(C(=O)NCc1c(CC)nn[nH]1)C N(C1CN(C(C2(C3CCC3)CC2(F)F)=O)Cc2ccccc21)C(C1CCC1)=O c1(CNC(=O)CC2CC(NC(c3cnnc(Cl)c3)=O)C2)cc(Cl)nc(Cl)c1 CC(C)(C)C(=O)OCCCC(=O)NC1CCN(S(C)(=O)=O)C1 c1(N(C2Cc3ccccc3C2)C)[nH]c(=NCC(C)(C)CS(C)(=O)=O)nc2scnc12 N1(C(C(C)SCCCC)=O)CC(F)CC1CNC(c1noc(CC)c1C)=O c1(CNC(=O)NC2CCCC2SC2CC2)cn(C2CC2)nn1 c1(CC(N2CCC(CNC(C3(C)CCCO3)=O)C2)=O)ccc(Br)nc1 N1(C(C2C3(CC(C)(C)C3)C2)=O)CCCC12CCN(C(c1sccc1Cl)=O)C2 N1(C(C(c2cccc(C)c2)=O)=O)CCC(NC(C2CCCN2C(C)C)=O)C2CC12 C1(C2CCCO2)(C(N2CC(NC(C(C)=CC)=O)CC3(C2)CC3)=O)CCCO1 CC(CCN(C)C)C(=O)NCC1CN(c2ncns2)CCO1 c1(OC)ccc(C(N2CC(NC(C3(N(C)C)CC3)=O)C3CC23)=O)cc1O Cc1cccc2cc(C(=O)N(C)CC3CCCN3C(=O)C#CC3CCC3)oc12 C(=O)(CS(C)(=O)=O)NC(C(=O)N(CCC)C)Cc1cc[nH]n1 N1(C(CC(=O)OCC)=O)C2CCC1CC(F)(CNC(=O)CCCCC(C)(C)C)C2 N1(CCNC(C2N(CC)CC2)=O)CCCN(C(c2cnnn2C)=O)CC1 C1(CCNC(C2CC(O)(CNC(CCc3n(C)cnn3)=O)C2)=O)CCCC2CC12 CN1N=C(C(=O)NC2CC3CC(C2)N(C(=O)CSc2cccs2)C3)CCC1=O N1(CC(=O)Nc2cnc(C(F)F)[nH]2)CCC(c2cn(CC3CCCC3)nn2)CC1 N1(C(C2N(C(C(C)C(C)(C)C)=O)CCC2(C)C)=O)C2CCC1CC(CO)C2 C(N=c1ccn(CC(=O)NCCC#N)c(O)n1)c1ccc(OC)c(C)c1C N1(C(c2ccccc2S)=O)CCC2(CCN(Cc3cccc(Cl)c3)C2)C1 c1(C(N2C(CN(C(C(C)NC(CC)=O)=O)C)CCC2)=O)cc(O)nc(O)c1 c12ccc(nc1)c(=O)[nH]c2=O.C1(C(=O)NC(CC2CC2)C2CCC2)(COC)CC1 C1(CNC(C2C(C)(C(C)C)C2)=O)CCN(C(c2ccccc2SCC#N)=O)CC1 c1(C(=O)NCC(CN(C(c2c(CC)nns2)=O)C)O)ccc(OC)c([N+](=O)[O-])c1 C(C(C(=O)OC)N(C(=O)C(CNN(C)C)c1ccccc1)C)OCC=C N1(C(C2ON=C(C)C2)=O)CC(NC(C2CC(C(F)(F)F)C2)=O)C(C2CC2)C1 N1(C(C(C)n2cncn2)=O)CCN(C(c2nncn2C2CC2)=O)CC1CO CCC(C(=O)NC1CC(N(C)C(c2ccc(C(F)(F)F)o2)=O)C1)n1cncn1 c1(SC(C)(C)C)ccc(C(=O)NC2(C)CC(NC(C3C4CCC3CC4)=O)C2)cn1 C1(C2CCCN(C(=O)C=C3CCC3)C2)(NC(CCC(=O)N(C(C)C)C)=O)CC1 Cc1cc(C(=O)NC2CC(CC(=O)NCC34CC(CCO3)C4)C2)cnc1O c1(SC)ccc2ncnc(N3CCC(N4CC(F)C4)CC3)c2c1 C1(OC)CC(C(=O)NC(C)Cn2cccn2)N(C(=O)C=CCN2CCC2)C1 CC1CN(C(=O)CC(CC2CC2)NC(=O)CC2CCCN(C)C2)CC(=O)N1 c1(C2C(C(=O)NC3C(NC(CCC)=O)CCC3)C2)ccc2c(c1)OCCO2 C1(CCNC(c2nc(C)n(C)c2)=O)CCN(C(=O)CS(=O)(=O)C2CC2)CC1(F)F C1(CNC(COC2(C)CCC2)=O)CCC(NC(=O)CC2CCCCO2)CC1 CC1C(C(=O)NC2C3CN(C(=O)CS(=O)(=O)CCO)CC23)=Cc2ccccc21 CC(C)C(O)CCN=c1[nH]c(=NC(C)CCC2CCCCC2)[nH]c2ccsc12 C(=O)(C1=NOC(C)C1)NC1(CCCNC(C2(OC)CCCSC2)=O)CC1 c1(C(N2CCN(C(c3c(SC)scc3)=O)CC(O)C2)=O)cccc2ncn(C)c12 c1(C(=O)NCCN(C(=O)Cc2nc[nH]n2)CCOC)cccc(C(F)(F)F)c1 c1(NC2C(=C)COC2)cc(-n2cccc2)cc(Cl)c1 C1(C(N2CC(O)(CCC)C2)=O)CCC(C2CC2)N1C(c1c[nH]c(C#N)c1)=O c1(C(=O)NCCN(C(C2CC2(COC)CC)=O)CC)ccc2c(c1)C1CCC2O1 c1(CN(CCCNC(c2c(C)nns2)=O)C(C)C)ccc(Cl)c([N+](=O)[O-])c1 c1(C(=O)NCCN(C(CC)C)C(C2CC=CC2)=O)ccc2c(c1)NC(=O)CS2 c1(C(N(C)C)=O)ccc(C(=O)NC2CC(C)(CNC(=O)CC34CC(C3)C4)C2)cc1 C(c1cc(C)ccn1)=CC(c1nnnn1C1CCC1)NCc1c(OC)ccnc1 N1(C(CCC(=O)OCC)=O)CC2CCCC(C1)N2C(=O)C(CC)SC c1(CC(=O)NCC(CNC(C(c2ccccc2)NC(N)=O)=O)F)ccc(O)cc1 n1(CC)nccc1C=CC(N1CC(NC(c2cc(C)oc2C)=O)C(O)C1)=O CCCCC(O)C(=O)NC1CCC(C(=O)Nc2cnc[nH]2)C1 c1(C(=O)NC2C(C)N(C(C3CC4(CSC4)C3)=O)CC2)cc2ccc(F)cc2o1 N12CCCC(C1)C2=O.N1(C(=O)OCC)CCC(NC(=O)C(=O)NCC2CC2)C1C Cc1cc(=NC(=O)CN(CC(C)NC(=O)CCC2CCC(O)CC2)C)[nH]o1 C1(C(N2CC(CNC(C3CC(C)(F)C3)=O)OCC2)=O)Cc2ccncc2C1 N1(C(CCCC#CC)=O)CCCCC(NC(c2ncnn2CC)=O)CC1 c1(SCC)ccccc1C(=O)N(C1CN(C(=O)CNC(=O)CCC)CC1F)C c1(C(N(CCCN(C(C(COC)OC)=O)C)C2CC2)=O)cccc(C)c1 c1(NC(C2(CC#C)CC=CCC2)=O)ccc2sc(S)nc2c1 C#CC(C)(C)C(=O)NCC1CCC1NC(=O)C(F)C(C)C N1(C(CCCC=C)=O)CCC2CCN(C(c3cc(CC4CCC4)c[nH]3)=O)CC2C1 CC(F)(F)CCC(=O)N1CC(NC(C2(C#N)CC2(C)C)=O)CC(O)C1 C1(NC(C2COCCO2)=O)CC(NC(C2CC(F)(F)CS2)=O)C(O)C1 CC1CCc2c(C(=O)NC(C)CNC(C3CC34CC(O)C4)=O)csc2C1 O=C1CCC(C(=O)N2CC3(CNC(C45CCCCC(F)(C4)C5)=O)CC2CO3)=NN1 C=CC1(CC(=O)NC(c2ncnn2C)C)CN(C(c2cnnn2C2CC2)=O)C1 C1(CCNC(Cc2c(C)cco2)=O)CC(F)(F)CN1C(=O)CCCC(=O)N(C)C c1(C(N(CC(CC)NC(CCNC(=O)OCC)=O)C)=O)cnoc1CC(C)C C1(NC(C2N(CC(C)C)CCC2)=O)CN(CC=O)CC1(C)C.C1CC1 c1(C(=O)NC(C)CNC(c2[nH]nnc2C2CC2)=O)c(O)ccc(Cl)c1F c1(C(=O)NCC2C(NC(C(N)=O)=O)CC2)ccc2ncccc2c1 N1(C(C(CC(=C)C)NC(c2c[nH]ccc2=O)=O)=O)CC2CCC1C(O)C2O CCC(C)CC(C(=O)NCc1ccncc1CO)NC(=O)C(=O)N(C)C C1(C(=O)NC(CNC(c2nc(C(C)C)sc2)=O)C)CC2(COCCO2)C1 N1(C(C(C)SCC)=O)CCC(CNC(c2cnncc2O)=O)C(O)C1 c1(C(=O)OC(C)(C)C)cc(F)c(C(=O)NCc2c(C(=O)OC)cccc2)cc1F c1(NC(c2nccc(C3(NC(=O)NC)CC3)c2)=O)cc(Cl)cc(OC)c1OC C1(CNC(=O)COCCc2ccccc2)CN(C(C2(F)CCOC2)=O)CC1(F)F CN1CC(=O)NC(CC(N2C3CCC2CC(NC(c2cnn[nH]2)=O)C3)=O)C1=O c1(OC)ncccc1C1CC1.C1(=O)C(C)N1.C12(CC1)CCCNC2=O Cc1ncc2n1CCN(C(C1CC(C)(NC(c3cccc4ccoc34)=O)C1)=O)C2 N1(C(=O)C2CC2)CC2CC1CN2C(=O)CC(=O)N(c1ncc(C(=O)OC)nc1)C c1(C(=O)NCCC2CCN(C(=O)CC3COCC3O)CC2)ccc2cncn2c1 c1(C(=O)NCCS(CCOC)=O)nn(-c2cccc(F)c2)c2c1CCCC2 N1(C(CCNC(C(C)(C)C)=O)=O)CC2CC1CN(C(=O)CCN1CCOCC1)C2 CCCC(CC)CCC(=O)N(CCCN(C)C(C1CCC(F)CC1)=O)C N1(C(C(F)=C(C)C)=O)CC(O)(CCNC(c2cnsn2)=O)C1 c1(C(=O)NC(C2CCCN2C(c2c[nH]c(C(F)(F)F)c2)=O)(C)C)c[nH]ccc1=O CC1(C)OC(=O)CC1C(N1CCN(C(=O)Cc2nc(C3CC3)cs2)CC1)=O CC(F)(F)C(F)(F)CC(=O)NCC1(C)CN(C(c2sccc2F)=O)CCO1 Cc1cc(=O)c(C(N2CCCCC2CCNC(=O)C(F)OC(F)(F)F)=O)c[nH]1 c1(CC(N2CC(C(=O)Nc3c(C(=O)NC)cccc3)C2)=O)ccc(Br)cc1I N1(C(C(N2CCOCC2)C)=O)CCC(F)(F)C(C(=O)Nc2cccnc2)C1 c1(C(N2CC(CC=C)(NC(=O)CSC)C2)=O)cnc(F)c(Cl)c1 N1(C(C=Cc2ccc(CC)cc2)=O)CCCC2(CCN(C(=O)CCSC)C2)C1 C(=O)(C(CC(F)F)C1CCC1)N(C1CC(NC(=O)Cc2nc(=N)[nH][nH]2)C1)C C(=O)(CCCC(=O)N1CC(CNC(c2conc2C2CCC2)=O)C2CC12)NCC CC1(F)CCCCN(C(=O)COCCNC(=O)CCCCC#N)C1 c1(C(N(CCNC(C(C)OCC)=O)CC)=O)ccc(F)c2ccccc12 c1(C(N2CCC(c3ccccc3)(NC(CCC=C)=O)C2)=O)cc(C)nc(C)c1 C1(CNC(c2cc(C(C)C)[nH]n2)=O)CCCCN(C(=O)C=CCn2cncn2)C1 C1(OC)CC(CNC(=O)CCCNS(C)(=O)=O)N(C(=O)CCCc2nccs2)C1 C1(NC(c2c(C)cco2)=O)CC2CC(NC(=O)C(F)CC3CCCC3)C2C1 n1(CC)nc(C(C)C)cc1C(=O)NC(C)CN(C(=O)Cn1cccn1)C CCCC(CCC)C(=O)NC1CC(NC(=O)CCn2c(C)ccc2C)C1 C(CC(C)C(=O)N(c1ccc(Cl)cc1)C)=CCC.C1(CC2CCCO2)C(=O)N1 N1(C(c2cccc(SCC#C)c2)=O)CCN(C(c2cc(C#N)c[nH]2)=O)C(C)C1 c1(C(N2CCC(NC(C(C(C)C)N3CCCCC3)=O)C2)=O)ccc([N+](=O)[O-])[nH]1 C1(C(N2CC(O)(CC(C)C)C2)=O)CC2C=CC1N(C(=O)CN1CCCCC1)C2 c1(OCCC)ncccc1C(=O)NCCNC(C1CCOC(C)C1)=O C1(C(N(CCOCCN(C(=O)Cc2cnsc2)C)C)=O)CCS(=O)(=O)N1 C1(CC)CCN(C(=O)CC2CC3(CCC3)C2)C1C(=O)N(CCC(F)(F)F)C Cc1cccc(C)c1CC(=O)NC1CCCC(NC(C23CC(CO2)C3(C)C)=O)C1 C1(CNC(C2(F)CN(C(C3CC(N(C)CC)C3)=O)C2)=O)CN2CCC1C2 N1(C(C=Cc2cncc(C)c2)=O)CC2(COC(CNC(=O)C(F)CC3CC3)C2)C1 CCCC(C)CC(=O)N(CCCCCCNC(=O)CCn1cccn1)C C(C(C)(CC(C)C)NC(=O)C1=NOC(C(C)(C)C)C1)NC(c1c(C)cc(C)s1)=O N1(C(CCC=C)=O)CCN(C(C2CC(=O)N(C(CC)CC)C2)=O)C2(CC2)C1 C#CCC(C)(C(=O)NCC(C)OCC=C)NC(=O)CC1OCCC1C c1(CC)cc(C)c(NCC(C2CCCC(=O)N2)(C)C)cn1 C(=O)(N=c1cc[nH]c(C)c1Br)c1ncc(-c2ccc(C)o2)cn1 c1(C(=O)NCC2N(C(C(CC)OC)=O)CC(F)(F)C2)ccc(F)c2ccccc12 N1(C(=O)C(F)n2ccnc2)CCN(C(c2ccc(=O)n(CCO)c2)=O)C2CCC12 c1(NC(C(=O)NC2CCCN(C(C(C)N3CCC3)=O)C2)=O)ccc(C#N)c(Cl)c1 N1(C(C(C)Oc2ccccc2)=O)CCOCC1CC(N1CC2CC2C1)=O CCC(C)C(C(=O)Nc1nnc(-c2nn[nH]n2)s1)N1CCCC1 C1(NC(C2CCC(=O)C2)=O)CN(C(=O)C=C2CN3CCC2CC3)C2(CCCC2)C1 C1(NC(CCC2(C)CC2)=O)CN(C(=O)Cc2ccc(F)cc2)C2(CCCOC2)C1 c1(OC)ccc(Cl)c(C(=O)NCC(C2CCCC2)NC(=O)CO)n1.C1C(=O)O1 Cc1cc([N+](=O)[O-])ncc1C(=O)Nc1ccc2c(c1)COC2 C=CC1CCCN(C(c2ccnc(CNC(c3ccsc3C#N)=O)c2)=O)C1 c1(OC)ccc(NC(=O)C(N2CCCC(c3n[nH]cc3I)C2)=O)c(OC)c1Br c1(C(N(CC)Cc2cc(F)ccc2F)=O)cc(C2=CCSCC2)n[nH]1 c1(C(=O)NCC2C(NC(C(C)c3ccco3)=O)CCCC2)cc(S(N)(=O)=O)c[nH]1 C1(C2CCCC2)(C(N2CCOC3CN(C(CCCSC)=O)CC32)=O)CCNC1=O N1(C(CCc2cc(C)no2)=O)CCN(C(C2(O)CCOC2)=O)CC(C)C1 C(C1CCN(C(c2ccccn2)=O)CC1)=CC(=O)NC1(C)CC(C)C1 c1(CNC(C2C(CCC)C2)=O)ccccc1CNC(C1CCCC12CC2)=O C1(NC(c2nc(C)c(C)s2)=O)CC2CN(C(=O)C(C)C3CCC3)CC2C1 N1(C(CSCC#C)=O)CCC2(C=C(C(=O)NCC(O)CC3CCCC3)C2)C1 C1(C(N2CC(NC(c3c(OCC)ccs3)=O)C(C)C2)=O)CCC2(CC1)CC2 CC1CCC(Cl)=C(C(=O)N(C2CC23CC3)C)C1 c1(C(N2CCN(C(C(CCC)C)=O)CC2CC)=O)cc(=NC)[nH]c2ccccc12 C1(C(=O)NC2CC(NC(C(Cc3cn(C)nc3)O)=O)C2)C2CCCCCC12 C1(NC(CCSC)=O)CN(C(c2ccc(C)c(-n3cccc3)c2)=O)CCC1C C1(CC(N2CCC(CCNC(C(C(C)O)C)=O)CC2)=O)CCCC2CCCCC12 C1(C(N(C2CCC2)CC)=O)CCCN1C(=O)CCOCC1CC1 C1(CNC(CC(C)OC)=O)CC(NC(c2ncsc2C2CC2)=O)C(O)C1 C(=O)(C(C(=O)NCC(=O)NCC(=O)NCc1cncc(CSC)n1)OC)OC Cc1cccc2c1C(NC(C1CCCN(CC(C3CCNCC3)O)C1)=O)C(=O)N2 c1(CC(=O)NCC(CC(F)(F)F)NC(C(C(C)C)O)=O)ncn2c1CCCC2 Cc1cccc(F)c1CC(=O)NC1(C)CCN(C(=O)CC(C)C)CC1 N1(C(CCCC)=O)CCCC2(CC(NC(c3sc(Br)cc3F)=O)CO2)C1 c1(C(C)=O)cc(C(=O)NC2CCC2NC(=O)Cc2nnc(O)s2)oc1C C1(NC(CCN(C)CC)=O)CCN(C(C2CC(C)(C)C2)=O)CC1C S(=O)(=O)(c1cc(C(F)(F)F)ccc1NC1C=CC(CO)C1)N1C(C)C(O)CC1 c1(C(N(CCCCN(C(C2C(C)OCC2)=O)C)C)=O)ccnc(-n2cccn2)c1 CC1C(NC(c2cnsc2)=O)CCCN1C(c1cc(-n2cccn2)ccn1)=O CN1CCN(C(c2occc2C2CC2)=O)CC1CNC(=O)C(c1cnn(C)c1)O c1(C(=O)NCC(F)CNC(c2ncnc(O)c2Cl)=O)cccc2c1NCCC2 c1(C(=O)NC2CC(NC(CSC)=O)C23CCC3)nnn2cc(C)nc(O)c12 Cn1cncc1CCNC(=O)C(Cc1cnc[nH]1)NC(=O)CC1CCCSC1 CC1=NOC(C(=O)NCC2(C3CCCCO3)CC2)C1C CCC(C)C(C(=O)NCCC1CCN(c2ncc(COC)cc2Cl)CC1)OC c1(C(N2CCC(O)(CN(C(=O)C=Cc3cnc[nH]3)C)C2)=O)ccsc1S(N)(=O)=O c1(C(=O)NC2CC(NC(C3C(C=C)CC3)=O)C2)ccc(-c2ccccc2)nc1O N1(C(C(CCCC)NC(=O)CCc2ccncn2)=O)Cc2c[nH]nc2C(C)C1 C1(NS(CC=C)(=O)=O)C=CC(=O)N=N1.C12CCCN1C(=O)C2 c1(C(=O)NC2CC(NC(C(C(C)C)OC)=O)C2)cc2cc(Cl)ccc2n1C C1(C(N(CC(CN(C(CC=C)=O)C)O)C)=O)CCCN1C1CCCCC1 C(CCC)(CCC)NC(C=CCC1(NC(CCC=CCC=C)=O)CCC1)=O c1(C(c2nnnn2C2COC2)NCCF)ccn(C(C)(F)F)n1 C1(OC)CC(CNC(C2(C)CS(=O)(=O)C2)=O)N(C(=O)CCCc2csc(=N)[nH]2)C1 C1(O)(CNC(=O)CC(O)C2CCCC2)CCCN(C(c2nncs2)=O)C1 c1(C(N2CC3(CCN(C(CC(=C=C)C)=O)C3)C2)=O)cnc2sc(C)cn2c1=O C(C(C)(C)C(=O)NCC(C1CCN(C(=O)C(c2cccnc2)O)CC1)O)N(C)C C(C)(CN=c1ccnc(NC(CC(F)F)c2ccccc2)[nH]1)OC C1(O)(CNC(c2c(CCC)nns2)=O)CCN(C(=O)C(N2CCOC2=O)C)CC1 c1(C(=O)NC2C3CCC(CN(C(C(CC)C)=O)C3)C2)cncc2c(F)cccc12 CC(C)C(O)CC(=O)N1CC2(CO)CC1(C(=O)NCC(c1ccccc1)O)C2 S(=O)(=O)(c1ccc(=NCCS(=O)C(C)(C)C)[nH]c1)NCCCC CC1CCN(CCc2cn(CCCC(=O)N3CCC3CC3CCCC3)nn2)C1 c1(NCC2COCC(C)O2)ccc(S(=O)(=O)NCc2csc(C(F)F)n2)c(Br)c1 c1(C(=O)NC2CC3(C2)CN(C(C2CC(C4CC4)C2)=O)C3)c(Cl)ccc2c1OCO2 c1(C(=O)NC2C3CC(NC(c4occ(C)c4)=O)CC32)cccc2ccn(C)c12 c1(C(=O)NCC2CCN(C(c3cn(CCC)nn3)=O)C2)cccc(S(C)(=O)=O)c1 c1(NC(C2N(Cc3cccc(OC)c3OC)CCOC2)=O)csc2ccncc12 C(=O)(CCCC(=O)OCC(=O)NCCSC)N1CCC(OCC#C)C1 C1(CNC(Cc2ccc(N)cc2)=O)CN(C(C2(C(N)=O)CC2)=O)CCCO1 CC(C)CC(CNC(=O)C(C)(C)Nc1nccs1)NC(=O)CSC1CCCCO1 c1(CNC(=O)NC(Cc2cscn2)Cc2ccccc2)noc(C(F)(F)F)n1 C1(NC(C(CSC)(C)C)=O)CC2CCC1N(c1nccc(CC(=O)OC)n1)C2 c1(C(N(C2CCCN(C(c3ocnc3C)=O)C2)CC)=O)cc2c(nn1)OCCS2 CN1CCCC(CC(N2CCC(C(C)(C)C)(CNC(=O)C(C)(C)CF)C2)=O)C1 C1(C(N2CCC(C#N)C2)=O)CCCCCN1C(=O)C=C1CCC1 c1(C(=O)NC(C)(CNC(=O)CCc2cnoc2)CO)ccc(C2CC2)cc1Cl c1(C(N2CCN(C(c3cc(F)cc(Cl)c3)=O)C(CO)C2)=O)cc(Cl)cnc1Br N1(C(CN(C2CCC2)C)=O)CC2CCC1CN2C(=O)CCC1CCCOC1 C=C(C)CC(C(=O)NCC=Cc1cccnc1)NC(=O)C(C)CCCOC Cc1occ(C(F)(F)F)c1CC(=O)NCC(C(C)C)NC(C1(CC(F)F)CC1)=O C(CC(C(=O)NCc1ccc(C)nc1)NC(=O)CC1CCCC1O)SC c1(C(=O)NCCC(C)N(C)C(C2C3CCCC23)=O)cnccc1N1CCOCC1 C(=O)(C(C)(C)C(O)C(C)C)N1CC(OC)(CNC(=O)C=Cc2cccc(F)c2)C1 C1(NC(C2=NOC(C)C2)=O)CN(C(=O)CC2=CCN(C)CC2)Cc2ccnn2C1 C1(C)CCc2ccccc21.C(C(C(=O)NCCN(C)CCOC)NC(C)=O)OCC N#CCCCCC(=O)N1CCCC(NC(C2(C(F)F)CC(F)(F)C2)=O)C1 N1(C(Cc2c(C)noc2Cl)=O)CC2CCC(C1CO)N2C(c1ccoc1)=O c1(NC2C(CC(=O)NC(C)C(=O)NC(=O)C(Cl)(Cl)Cl)C(O)C2)ccc(O)cc1F C=CC(CC)C(=O)NC1CCC(CC(=O)NCC(C)(O)C(F)F)C1 C1(C(=O)NC(CO)C2(O)CC2)(CO)CCN(C(C2CN(C3CC3)C2)=O)C1 c1(NC(C(C2CCCN(C(c3scnc3C(F)F)=O)C2)C)=O)ncccc1O c1(-c2nc(C3CCC3)nn2C(C)C(C)(C)C)n[nH]c2c1CC(C)(C)CC2 CCCC(CCCS(C)(=O)=O)C(=O)NC1CC(CNC(=O)C2=NOC3(CCC3)C2)C1 C(c1ccccn1)=CC(N1CCC(NC(=O)Cn2cnc(=N)[nH]2)C1)=O c1(-c2n(CCOC)c(N3CCOC(C(C)(C)C)C3)nn2)nccn2cccc12 c1(C(=O)NCC2C3CN(C(C4CC45CC(O)C5)=O)CC23)cn2c(n1)CCCC2 Cc1ccc(-c2ccc(C(=O)N(C)CC3CCCN(C)C3)o2)cn1 C1(CN(C(C2C(C)OCC2)=O)C)CCCCN1C(=O)C(N1CCOCC1)C c1(C(C(=O)NCC(=C)C)N(CC(=O)OC)CC)cc(Cl)ccc1Cl.C1CN1 CCCC(C(=O)N(CC(N1CCCC1CC(=O)OC)=O)C(C)C)N(C)C Cc1cc(C(=O)NCC(C)NC(c2cnn(C)c2)=O)cs1 N1(C(c2snc(C)c2N)=O)CCC2CCN(C(c3coc(O)n3)=O)C2C1 CC12CC(C(N3CC(=C(F)CNC(=O)CCC4CC4(C)C)C3)=O)(C1)C1(COC1)O2 c1(C(=O)NC2C(NC(CN(CC)CC)=O)CCOC2)ccc(NC)c([N+](=O)[O-])c1 n1(CC(N2CC(N(C(C(CC)OC)=O)C)C3(C2)CC3)=O)c(C)nc2ccccc12 c1(NC(C2CC(F)CN2C(c2ccccn2)=O)=O)cc(F)c(Cl)cn1 CC(C)(CO)C(O)C(=O)NC1CCCOC1 C1(C(N(CC(C)NC(=O)Cc2cncs2)C)=O)CC12C1CC3CC(C1)CC2C3 n1(CC(=C)C)c(N2CCOC(C(N)=O)C2)nnc1-c1ccnc(C)c1 N1(C(c2n(C)ncc2[N+](=O)[O-])=O)CCCC2(CCN(C(=O)C(N)=O)CC2)C1 C1(C(=O)NC2C(CCOC)CCC2)CCC(C)CN1C(=O)Cc1cc[nH]n1 CC1OC(C)(C)OC1(C)C(=O)NCC1(F)CN(C(c2ccnnc2O)=O)C1 c1(C(N2CC(NC(Cc3cc(C)no3)=O)C(C#N)C2)=O)cnc2cc(Cl)ccn12 C(N=c1ccc(Br)c(S(=O)(=O)NC2CC3CCCC3C2)[nH]1)c1ccc(C)nc1 c1(CC(=O)NC(c2cc(Cl)sc2Cl)C)c[nH]c2ccncc12 C1(COC)CC(CNC(=O)CCC2(O)CCC2)N(C(=O)CCCn2cccn2)C1 c1(C(C)NC(C2NCCN(S(CC(=O)OC)(=O)=O)C2)=O)cc2ccccc2o1 c1(C(=O)NCCSc2ccc(OCCOC)cc2)cc2c(C)nn(CCCl)c2s1 c1(C(=O)OC)no[nH]c1=NC(=O)CC1CCN(C(=O)CC2CCCC2)C1 c1(NC(=O)Nc2c(C(=O)OC)cc(Br)cc2C)cc(C)c(F)cc1Br N1(C(=O)CCCCC2CC2)CCC2CCN(c3nc(Cl)ncc3C3CC3)CC2C1 C1(C(=O)NC)CN(C(=O)CCCC2CCCO2)CC1c1ccc(C)cc1 CCCC(C(=O)NC(CCN(C)C)C(=O)N1CC(N2CCC2)C1)OCC C1(N(C(c2n(CCC)nc(C)c2)=O)C)CC2CCC(C1)N2C(c1cc(Cl)c[nH]1)=O c1(C(=O)NCC(C(CC)CC)OC)cc2ccc(F)cc2nc1O N1(C(C(=Cc2cccs2)C)=O)CCCC2(CCN(C(C3CCCC3O)=O)C2)C1 c1(C(=O)NC(C(C)C)CCN(C)C(c2cncs2)=O)cc2c(F)cccc2[nH]1 O(NC(=O)N=c1[nH]nc(C)n1C1CC1)C(CC)Cc1ccccc1 CC12CC(NC(=O)C=C(Cl)Cl)(C1)C1(CN(C(c3cccc(CO)c3)=O)C1)O2 C(=O)(C(CC(C)(C)C)OC)NCC1(COC)CN(C(=O)Cc2ccc(C)nc2)C1 c1(C(N2CCC(C(C)(C)CNC(C3CC34CC4)=O)CC2)=O)ccc(Br)cc1N Cc1cccc2c(C(N3CC4(NC(C5CCCCC(=O)N5)=O)CC3C4)=O)n[nH]c12 CC1(NC(=O)CN(C(=O)C=Cc2ccco2)CC2CC2)CCOCC1 Cc1cccc2c1OCCC2Nc1nccc(N2CCC(n3cccn3)C2)n1 c1(C(=O)NC2(CC(N3CC(C(N(C)C)=O)C3)=O)CCC2)cnc(=N)[nH]c1 c1(C(Cc2ccccc2)NC(Cc2n(CC)cnc2)=O)ccccc1Br C1(NC(c2ccc(=N)[nH]n2)=O)CC2(C1)CN(C(C1(O)CC1)=O)C2 N1(C(C2(N(C(C(N3CCCCC3)C)=O)C3CC3)CC(O)C2)=O)CC2CN(C)CC2C1 CC1CN(C)CC1NC(=O)CCN(C(=O)Cc1cnns1)C C1(C)(C(N2CC(NC(c3c(C)cc(F)cc3)=O)C(C)(C)C2)=O)CCC(C)C1(C)C N1(C(COC)=O)CC(CNC(C2(Br)CC2(F)F)=O)(OC)C1 CCCCC(CC)CC(=O)NCCCC(C)(C)C(=O)NCC(O)CC1CCCC1 CC(C(C)C(=O)NCc1nnc(O)o1)NC(C1COCC(C)O1)=O C1(F)(C(=O)NC(c2cccs2)(C)C)CCN(C(=O)COCC2CCOC2)C1 c1(OC)cc(F)c(CNC2CN(C(c3csc(C)n3)=O)CC2C)c(F)c1 c1(C(N2CC(F)(C(=O)OC)C2)=O)ccc2sccc2c1 n1(CCN(CCCC)CC)c(N(c2cccc(CC3CCCO3)c2)C)nnc1C c1(C(=O)NCC2N(C(CCc3ccc(C)s3)=O)CC2)coc2c1CS(=O)(=O)C2 C(=O)(C1=CC2(CCOCC2)C1)NCC1N(C(=O)OC(C)(C)C)CCC(C)(C)C1 N1(C(C(c2c(C)n[nH]c2C)C)=O)CCCC2CN(C(=O)Cc3n[nH]c(=N)s3)CC12 c1(CN(C(c2nccc(OC)c2)=O)C2CC2)cc2ccccc2o1 c1(C(N2CCC(C(C)(C)NC(C(=O)N(C)C)=O)C2)=O)ccc(S(C)(=O)=O)o1 c1(NC(CC)CSC)ncnc2cc(Br)c([N+](=O)[O-])cc12 C(CNC(=O)C(COC)Oc1ccccc1)(C(C)(C)C)NC(CN(C)CC)=O C(=O)(N=c1ccn(C2CC2)[nH]1)C1CCCC(NC(C(CCC)F)=O)CC1 N1(C(CN(CC)CC)=O)CCCC2CN(C(=O)C(C)=CCSC)CCC12.C(C)(C)(C)O c1(NCC(=O)NC2(C(NOC(CC#C)C)=O)CCC2)nn(C)cc1C N1(C(CC(CCC)C)=O)CC2=C(C1)CN(C(=O)CCCCNC(N)=O)C2 CCC(CC(=O)NCc1nnnn1C)NC(c1cc(C2CC2)[nH]n1)=O C(=O)(C(C(F)(F)F)NS(=O)(=O)Cc1ccccc1SCC)OCC C1(OC)CC(C(N2CCN(C(C)CNC(=O)CC3(C)CC3)CC2)=O)CC1OC C(C(F)(F)C(=O)NCC(O)CNC(c1cccc(-c2cscn2)c1)=O)OC CCCCC(C(=O)NC1CC(CNC(c2cc(F)cc(F)c2)=O)C1)N(C)C C1(C2CCN(C(c3conc3C3CC3)=O)C2)(NC(=O)C=C(Cl)Cl)CC1 C1(NC(c2ccc(C3(F)CC3(F)F)cc2)=O)C2CN(C(=O)Cn3cnnn3)CC12 C1(N(CC#C)C(c2cc(C)co2)=O)CCN(C(C2CC(C)CO2)=O)CC1 CN1CC(=O)NCC1C(C=CC(N1CCOCC(CNC(=O)C(F)(F)F)C1)=O)=O c1(NC(c2ccc(NCc3cccc(C)n3)cn2)=O)ccc2ncn(C)c2c1 C1(NC(C)CCc2cccnc2)C2CCCC1CC2 CCC(CC(C)CO)NC(=O)CCCNC(C1(O)CCCC1)=O c1(NCC(=O)NCC2(O)CN(C(C(=O)NCCNC(C)=O)=O)C2)ccc(F)cc1 C1(CNC(C2CCN(CC)C2)=O)CN(C(=O)CCc2cncc(O)c2)CCCO1 C(C)(C(C(=O)NC1CCCC1CF)C(C)C)NC(c1n(CC)nnc1)=O c1(C(=O)NCC(C)N(C(c2n[nH]cc2C)=O)CC)oc(-c2ccccc2)nc1C C1(NC(c2c(C)coc2)=O)C2CC3CN(C(c4cnc(Br)s4)=O)C1C3C2 Cc1cccc(F)c1C(N1CCC(N(C(=O)CCc2cc[nH]n2)C)CC1)=O C1(NC(C(CC)CC(C)C)=O)CCC2(CC1)CN(C(c1csnc1C)=O)CCO2 n1(CC(=O)NC(CC)CN(C(=O)C(F)OC)CC)nc(C)c(Cl)c1C C1(C(=O)NC(CCC)CO)C2CCC(C2)C1NC(c1nc(C)oc1C)=O C#CCC(C(=O)NC1(CO)CN(C(c2sc(N3CCCC3)nc2Cl)=O)C1)C1CC1 C1(C(=O)NCC2CCCN2C(=O)Cn2cc(Cl)cn2)CC(C(F)(F)F)(OCCO)C1 C1(CNC(Cc2c(C)n(C)nc2)=O)CC2(CCN(C(c3cc(Cl)ns3)=O)C2)CO1 C12(n3cccn3)CCN(CC1)CC1(Cl)CCN1C2=O.C(=O)(CCCC(C)O)OC C1(O)(C(C)NC(=O)C=C2CCCC2)CCN(C(=O)CC(C)(C)O)C1 N1(C(C(COC)COC)=O)C(C)CC2CN(C(=O)COc3ccc(Cl)cc3)CC12 c1(C(=O)NC2CN(C(C3CC3C(N)=O)=O)C3(CCC3)C2)c[nH]c2cccc(F)c12 C1(CNC(C2(COC)CC=CC2)=O)CC2(C1)CN(C(c1cncc(Cl)c1)=O)C2 Cc1nc(CC(C)C)sc1C(=O)NCC(C1CCCC1)NC(=O)CC1COC(=O)C1 N1(C(c2cn(CCSCC(=O)O)nn2)(C)C)CCS(=O)(=O)CC1 c1(C(=O)NCC(C)CNC(C2(Cl)CC2(C)C)=O)ccc([N+](=O)[O-])c(O)c1 n1(CC)nc(C)cc1C(=O)N(CC(=O)NCCc1nc[nH]n1)C1CC1 c1(NC(C2C(NC(C=CC(C)C)=O)CCC2)=O)cccc([N+](=O)[O-])c1F CN(C)NC(=O)CCC(=O)NC(CC1CC1)C(N1CCC(N=[N+]=[N-])C1)=O c1(OCC)cncc(CNC(C2CCCCC2NC(C2OCCC2C)=O)=O)c1 N1(C(C(C)(C)OC(C)=O)=O)CC2CCC(C1)C(NC(=O)C(C)C(C)S(C)(=O)=O)C2 C12(C(=O)NCC3(CNC(C4OC5CCC4C5)=O)CC34CCC4)CCCC(CO1)C2 Cn1cc(C#N)cc1C(=O)NCC(C)(O)CNC(c1csc(C2CC2)n1)=O N1(C(c2c(CC)csc2)=O)CCN(C(c2cc(C)c(Br)o2)=O)C2CC12 CCCC(C(=O)OC)C(=O)NC(CC(=O)N1CC(OC(F)F)C1)C(F)F c1(C(=O)NC(c2ccc(OC)cc2)C)cccc(Sc2c(Cl)ccnc2Br)c1Cl CC1CN(C(=O)CCC2(C)CC2)CC(C)C1NC(=O)Cc1n[nH]c2c1CCCC2 C(CC)(CCCC(=O)N(CCCC)CCCC)NC(C(C)OCCC=C)=O C1(C(=O)OC)C(F)(F)C12CC(C(=O)NCCC(C)(C)NC(c1coc(C)n1)=O)C2 C1(NC(CC=C=C)=O)CC(CNC(C2CN(c3nnnn3C)C2)=O)C1(C)C C1(C2C(NC(C3CC(C)(O)C3)=O)CCO2)CCN(C(c2cccc[n+]2[O-])=O)CC1 C(c1ccc(=N)[nH]c1)=CC(=O)N(CC(=O)O)C.N1(C2(CC(=O)N)CC2)CCCC1 C1(O)(CCNC(C(CCC)N(C)C)=O)CCN(C(c2ccsc2Cl)=O)CC1 N1(C(C(C)=C(CC)C)=O)CCCC(C)(NC(c2cncc(OC)c2C)=O)C1 C1(CC)CCC(C(=O)NC(C2(C(=O)NCCCCSC)CC2)C)O1 c1(CNC2CC(C(N(C)CC3(C#N)CC3)=O)C2)sccc1Cl C1(C(=O)N(C)CC=CC(=O)NC(c2cscn2)CO)(OC)CCSC1 C1(C2CCCN(C(=O)COC3CC=CC3)C2)(NC(=O)Cc2cnoc2)CC1 Cc1cnc(NC2CN(C(C3(C)CNC(=O)C3)=O)CC23CCC3)nc1S(C)(=O)=O CC1CN(C(C2COCC2NC(C2C3CCC(F)(F)C23)=O)=O)CC(C)(C)C1 C1(NC(C(C(C)C)S)=O)CCOC2(CCN(C(=O)C(F)(F)c3ccco3)CC2)C1 c1(C(=O)NN2CCCC2C(=O)NC2C(SCC)C2)coc2cc(C)c(C)cc12 c1(-c2ccc(CNC(c3cncs3)=O)s2)ccc(F)cc1 C1(C(=O)NC2(COC)CC2)CCC2CCC1N2C(C1CC(C(C)C)C1)=O c1(OC)cnc(C(=O)NCCOC2CCN(C(=O)C=Cc3nnn(C)n3)C2)cn1 Cc1nn(CC(=O)NC(C)C(C)NC(c2ccc(F)c(O)c2)=O)cc1[N+](=O)[O-] c1(C(c2n(CC=C)nnn2)NCc2cnc(C3CC3)s2)cc(Cl)sc1C N1(C(=O)C=CCN2CCOCC2)CC2CCN(C(C3CCCCC3O)=O)C2C1 C1(C(=O)NCCOCCCNC(c2ncccc2O)=O)CC2(CO1)CC(F)(F)C2 C(C(=O)N(C)CC1CCN(C(c2sc(C(C)(C)C)nc2C)=O)CC1)(C(C)C)OC N1(C(C2CCC(NC(CC)=O)C2)=O)CCC(C2CN(C(=O)C=CBr)C2)CC1 C1(NC(c2cccnc2)=O)CCCC12CN(C(c1csc3nnsc13)=O)C2 c1(C(=O)NCC23CC2CN(C(c2ncc(Cl)cc2Cl)=O)C3)c[nH]c2ncccc12 N1(C(C2(CC)CC2)=O)CCC2(CCN(C(=O)CC34COC(C(=O)OC)(C3)C4)C2)C1 CC1CN(C(=O)CN2CCC2)CC1CNC(c1cccc(OC(F)(F)F)n1)=O c1(C(=O)NCCCN(C(C)C)C(C2COC(=O)N2)=O)cccnc1O CCCC(C)(CCC)C(=O)NC1CCCC(NC(=O)Cc2cc(C3CC3)no2)C1 c1(C(N)=O)ccc(C(=O)NCC2CCCN2C(C2(c3cccs3)CCCC2)=O)o1 N1(C(c2c(OC)cc(OC)c(Br)c2)=O)Cc2c[nH]nc2CC(C)C1 CC(C)C(C)C(CNC(C1(C2CC2)CCC1)=O)NC(=O)Cc1cc(F)ccc1F CC(CC(=O)NC1CCCN(C(c2cnc(C3CC3)s2)=O)C1)C(C)(C)C C(=O)(CCCCc1ccccc1)NC(C1CN(C(C(N2CCC(C)C2)=O)=O)C1)C C1(C(=O)NC(C)C(N2CC(CO)C(O)C2)=O)CC2C(C1)C2(C)C C(=O)(C(CC(F)F)NC(=O)COC1(C)CCC1)NC(C1CCOCC1)C N1(C(CCCC#CC)=O)CC2CC(C(N3CCC(O)C3(C)C)=O)C(C2)C1 N1(C(C(=O)NCCNC(C(C)C)=O)=O)CCCC([Si](C)(C)C)C1 c1(C(=O)NC23CCC2CN(C(C2CC24CCC4)=O)C3)cc(Cl)c(C(F)F)cc1F C(=O)(CC(F)(F)Br)NC(CNC(C(CC)c1ccccc1)=O)(C)CO c1(OC)ccc(C(N2CC(CNC(c3nncn3C)=O)C(C)C2)=O)cc1 C=C1CC(C)(C(=O)NC2CC(NC(=O)C(O)Cc3ccccn3)C2)C1 C1(CN(C(=O)CC2CCN(CC)C2)CC)CCOC1CNC(=O)OC(C)(C)C C(C(C)C(=O)NOCCN(C)C)SC.C(CC1C(=O)O1)NC(C)=O C1(C)(C(=O)NCC(C)(C)NC(c2cc(COC)no2)=O)CCC(C)=C(C)C1 c1(C(=O)OC(C2CC2)C2CC2)cnn2c1S(=O)(=O)CC2.c1(C)ccccc1 C#Cc1c[nH]nc1C(N1CCC(NC(=O)CCc2cn(C)cn2)C1)=O N1(C(C(C)Oc2ccccn2)=O)CC2CCN(C(=O)C3=CC(C)(C)C3)CC2C1 C1(C(N2CCN(CCNC(c3ccsc3Cl)=O)CC2)=O)SC2C=CC1CC2 CC(C)(C#N)CS(=O)(=O)NC(c1cnc2sccc2c1)=O C(C)CC(C)CC.C=C1CC(C(=O)N(CC)CC)(CNC(=O)C=CCOC)C1 c1(C(=O)NC2C(C)N(C(=O)CC3CCC3)CCC2)nccc2c(Cl)cccc12 N1(C(C2(n3cccc3)CCOCC2)=O)CC(OC2CCC2)C2(CC2)C1 C1(CC(=O)N(CCCCNC(c2csc(C(F)F)c2)=O)C)CCCCC1F c1(C(C)(C)C)noc(CCCC(=O)NCC2(O)CC(NC(C3(O)COC3)=O)C2)n1 C(C(C)CC(=O)N1CCCC1CC(N)=O)NC(c1cc(C)sn1)=O C(CC(=O)NCC1CCCOCC1)(C(C)(C)C)NC(C(=O)NC(C)C)=O C#Cc1ccc(C(=O)NCC(O)CN(C(=O)C(O)C(C)C)C)nc1 C1(C(=O)NCCN(CC(C)O)C(=O)CNc2cccnc2)CCCCNC1=O C1(C(=O)NCC2(CC)CCC2)C(C2CC2)CCN1C(c1ccnc(C)c1N)=O N1(C(=O)CCc2cnco2)CC2CC1CN2C(c1cccnc1O)=O N1(c2nnc(C#N)s2)CCCC12CCN(c1cccnc1)CC2 N1(C(Cc2c(C)cccn2)=O)CCC2CCCC12C(=O)NC(C1CCOC1)C C1(C(CNC(=O)CC(=C)Br)(C)C)CCN(NC(C2C(=C)C2)=O)CC1 C(=O)(C(CC(C)C)NC(N)=O)N(CCOCCN(C(CC(=C=C)C)=O)C)C c1(C(N2CC3(CCC(C(N)=O)O3)C2)=O)sc2ncccc2c1Cl Cc1c(NC(=O)CC(C)CNC(C2CCCCCCC2)=O)cccc1Cl C1(CNC(C(C)OC)=O)CCC(F)(CNC(=O)C(O)Cc2ccc(F)cc2)CC1 C1(NC(c2c(C)onc2-c2ccccc2)=O)CCN(C(C2(F)CC2C)=O)CC1F CC1(C)CN(C(c2csc(C(F)(F)F)n2)C(=O)NCC2(O)CCCCC2)CCC1O N1(C(c2nnc(C)s2)=O)CC(CCNC(=O)C(F)=C2CCCC2)OC(C)C1 C1(NC(C2(C)CC2)=O)Cc2ccccc2N(C(=O)CSCc2cccs2)C1 c1(C(=O)NC2C3(CN(C(c4cccc(C)c4F)=O)C3)CC2)ccn2nccc2n1 Cn1ncc2c(NC3CCN(C(=O)C(c4cscn4)N(C)C)CC3)ncnc12 N1(C(C(CC)F)=O)CCC2(CCCCN(C(c3cccc([N+](=O)[O-])c3Cl)=O)C2)C1 C12(CNC(CCNC(=O)CO)=O)CC(CNC(=O)CSC3CC3)(CO1)C2 Cc1ncn(O)c1C(=O)NCC1CCC(CN(C(C2C3CC4C(C3)C24)=O)C2CC2)CC1 N1(C(C2CC(=C)C2)=O)CC2(C1)SCCC2NC(c1ccncc1Br)=O C1(NC(c2c(C)n[nH]c2)=O)CC2CC(C1)N(C(c1cc(O)nc(C3CC3)n1)=O)C2 CCC(CC(=O)NCc1ccc(C(=O)NCCSCC(C)C)s1)SC O=S1(=O)CCC(S(=O)(=O)Nc2cc(Cl)c3c(c2)OCCCO3)CC1 C(=O)(C1CCCn2c(C)cnc21)NC(CC)CNC(c1cc2ccoc2cc1F)=O c1(C(N2CCC(N(C(=O)CC3(CO)CC3)C)C2)=O)ccc(F)c(F)c1 C1(CNC(C2N(CC)CC2)=O)CN(C(=O)C(C)c2cccs2)CCN1C c1(C(=O)NC2(CNc3ccc([N+](=O)[O-])cn3)CCCC2)cccc2c1CCOC2 N1(C(C(N2CCC(C)C2)=O)=O)CCN(C2CCOC2)C(=O)C1 Cc1cc(C(=O)N(C)CC2CCCN2C(c2nnn(C(C)C)c2C)=O)c[nH]c1=N c1(C(=O)NCCN(C(C(C(C)C)C)=O)C2CC2)c[nH]c2cccnc2c1=O N1(C(c2c(C)cnn2C(C)C)=O)CCN(C(c2cscc2C#N)=O)CCC1C C1(c2cccc(NC(C(N3CCN(C)CC3)=O)=O)c2)CNC(C)(C)CO1 C(=O)(CC(C)CC(F)(F)F)NCC(C(C)C)NC(C1ON=C(CC)C1)=O C1(NC(C(C)(F)F)=O)CC2CCC1N2C(c1ccc(Nc2ncccn2)cc1)=O Cc1cnc2c(cnn2CC(=O)NC23CCN(C(=O)C=CCO)CCC2C3)c1 C(=O)(CC(C)CC(C)C)NC1(CC=C)CCCN(C(=O)CCc2cccnc2)C1 C(C(C)(C)CC(=O)NCC1(n2nccn2)CC1)OC.C12CCCN(C1)C2 C1(CNC(CC(C)OC)=O)CCCC2(CN(C(c3nnccc3C)=O)C2)O1 c1(C(N2C3CN(C(C(CCC)(C)C)=O)CC2CC3)=O)cc2c(cc1Br)OCO2 C12(CNC(c3cc(CC)[nH]n3)=O)CCC(C1)C(=O)N2.C12(CCC1)C(=O)N2C1CC1 C1(C(=O)NC2CN(S(CC=C)(=O)=O)CC2F)CCc2cccc(OC)c2C1 N1(C(C(C(C)C)SCC)=O)CC2(CC(CNC(c3ccc(F)c(C)c3)=O)C2)C1 C1(C(N2CC(C)(OCC(=O)N(C)Cc3cccs3)C2)=O)(OC)CCC(C)C1 C(=O)(C(CC)C(C)C)NC(CCC)CNC(C1CCCC1)=O Cc1c(C(=O)NCCCCNC(=O)COC2CCCC(C)C2)c(C(F)F)nn1C N1(C(CCCOCC)=O)CCC(CNC(c2ccn(C3CC3(F)F)n2)=O)C(C)C1 C(=O)(C(F)(F)C(F)F)NC(CC(C)NC(=O)CSCc1ccc(F)cc1)C C(CC(CO)NC(C1(C(C)NC(=O)Cc2ccnn2C)CC1)=O)=CC c1(C(=O)NC2CCC(CCNC(=O)CC3CC3)C2)ncc(Cl)cc1O Cc1csc(C=CC(=O)NC(C)CCCCNC(=O)CCc2nc(C)cs2)n1 S(=O)(=O)(c1cccnc1NCc1ccc(=N)[nH]c1)NC(CC)CC(C)O C(=O)(C(C)S(=O)(=O)C(C)C)NC(CC=C)CNC(c1ccc(N(C)C)nn1)=O Cc1csc(=NCC(=O)N2CC(CNC(C3CCCSS3)=O)CC2C)[nH]1 N1(C(c2cccc(SC)c2)=O)CC2CC(NC(C3(CCF)CC3)=O)C2C1 C=C=CCCC(=O)NCCN1CCN(C(=O)CCc2cc(C)no2)CC1 C(=O)(C(C)C(CC)CC)N(CCCC(=O)NCCNC(=O)OC)C C(=O)(C1CCc2nccn21)N1C(CNC(c2cccc(F)c2Cl)=O)CCC1 N1(C(C2(CNC(C3CCCN(C)C3)=O)CC2)=O)CCC2(CC1)CC(O)CO2 C=CCC(C)(C)C(=O)N1CC(N(C)C(C23CCOC(C)(C2)C3)=O)C2(CC2)C1 C(C)(C)(CC(=O)NCC1CC(F)CN1C(=O)Cc1csc(NC=O)n1)SC CC1CCCC1C(=O)NCCCOCCNC(c1ccnn1C(F)F)=O C1(OC)CN(C(C2OCCC2(C)C)=O)CC1NC(=O)Cc1csc(NC=O)n1 C(=O)(C(F)C(C)CNC(c1cccc(OCC(F)F)n1)=O)N(CC)CC n1(C(C)C)ncc(C(N2CC(O)(C(F)C(=O)NCC(C)N(C)C3CC3)C2)=O)n1 C1(NC(=O)NC(c2ccc(Br)cn2)COC)CCNC(C(F)(F)F)C1 C12(CNC(=O)COC(F)F)CN(C(=O)Cc3cscn3)CC(F)(C1)C2 CCC(O)C(C)(C)C(=O)NCC(O)CN(C)C(c1c(C(C)C)n[nH]c1C)=O C(=O)(C1CCCc2ccccc21)NCC(N(C(=O)CN1CCCC1=O)C)C1CC1 C1(CC(=O)NC2(C)CC(NC(C(C3CCC(C)CC3)CC)=O)C2)CCCCCC1 N1(C(=O)Cn2cc(F)ccc2=O)CC2C3CCC(C2C1)N(C(=O)C(F)F)C3 C1(c2nc(CCC)[nH]n2)CCCN(CN2CC(C(=O)OC(C)(C)C)CC2=O)C1 C12(CNC(C3CCC(C(F)(F)F)O3)=O)CC(CNC(C3CCCO3)=O)(CO1)C2 N1(C(C2CC(=C)CN2C(c2cc(Br)c(O)c(Br)c2)=O)=O)CCC2(CCOC2)CC1 N1(C(C2CC2c2ccccc2)=O)CCC12CCN(c1ncc3[nH]ncc3n1)CC2 C1(C2CN(C(=O)Cc3cc(F)ccc3Cl)C2)(NC(C2CCC=CCC2)=O)CC1 c1(C(N2CCCC2c2ccc(C)nc2)C(=O)NCCC)ccc(OC)nc1OC C(=O)(C(C(=O)NC1CCC(N(C(=O)C(N)=O)C)CC1)C1CC1)OCC N1(C(c2nc[nH]n2)=O)CC(NC(C2(c3cncc(Br)c3)CC2)=O)C(F)C1 c1(OC)ccccc1-c1noc(CN(C(C)CNC(c2cnc(C)s2)=O)C)n1 CCC(CC(=O)N1CC(CO)(NC(=O)CC2(O)COC(C)(C)C2)C1)C(F)F c1(OC(c2c(OCCC)cc(C)cc2)=O)cc2c(nn1)CCCC2 n1(C(CC)CC)nc(C(=O)NC2CC(CCNC(c3ccoc3Cl)=O)C2)cc1C C1(CC)(CC)CC(NC(=O)C(C)(C)n2cc(Cl)cn2)CN1C(=O)C(C)SC C1(C(N2CC(Cn3cc(C(O)(C4CC4)C4CC4)nn3)C2)=O)C2CCCCCC12 C(C(=O)NCCCN(C(C1CC2CC2C1)=O)C1CC1)(C(C)C)NC(COC)=O C1(CNC(CC2C(C)CCC2)=O)CCCN(C(C23CC(C)(CO2)C3)=O)CC1 N1(C(C2CC(C)N(C)C2)=O)CC2CC(NC(c3ccn(C)c(=O)c3)=O)C(C2)C1 c1(NCC)cccc(C(=O)NCC(N2CCN(C(=O)C(C)N(C)C)CC2)C)c1 c1(NCC23CC(NC(C4CCC(c5ccccc5)O4)=O)(C2)C3)ncccc1CO c1(C(N2CCN(C(CC(CC)C3CC3)=O)C(C)C2)=O)ccnc2ncc(C)cc12 C1(NC(C2(C)C(C)CN(C(C3CCCC3)=O)C2)=O)CC2CC1OC(=O)N2 C1(NC(=O)CCN2CCC(O)CC2)CC(O)CN(C(=O)CSC2CCS(=O)(=O)C2)C1 C1(CNC(C(C2CCC2)OC)=O)COCCN(C(c2ccc(F)nc2)=O)C1 CC1CC(NC(=O)CCc2ccc[nH]2)CN1C(c1occc1Br)=O C1(C(N2C(C(=O)OCC)CC(F)(F)C2)=O)CC2(C1)CC(C)(C)C2 CC1CC(=O)NCCN1C(=O)CC1CCCC1NC(c1nnsc1N)=O n1(CCC)cc(C(=O)N(CC(CC)NC(c2ncc(F)cn2)=O)C)c(C)n1 Cc1sccc1C(=O)NCCCC(=O)NCc1noc(C(N)=O)n1 N1(C(CN(C)C)=O)CCc2cc(-c3cc(F)ncc3F)ccc2C1 CP(C)(=O)C1CCCCC(Nc2ccc(Br)c(C(F)(F)F)c2F)C1 C1(CNC(CCN(C(C)=O)C)=O)CN(C(C2CC2(Cl)Cl)=O)CC2(CCC2)O1 c1(C(=O)NCC2C(NC(CN(CCC)C)=O)C2)cc2c(nc1O)C(C)(C)CCC2 c1(C(=O)NC2CCN(C(COC)=O)CC2C)ccc(C2=CCOCC2)cc1 c1(COC)nc(C(=O)N(C2CCC(NC(C3(CC(C)C)CCCC3)=O)C2)C)co1 Cc1ccc(CN=C(NCc2c(C)noc2C)NCC2CCCCO2)c(C)c1 c1(-c2cnc(C)s2)ccn2ncc(C(=O)Nc3cc(C)ccc3[N+](=O)[O-])c2c1 c1(C(N(C(C)CNC(C2COC(C)C2)=O)CC)=O)cnc(OCCOC)cn1 S(=O)(=O)(c1ccc(Br)c(Cl)c1)NC1(C#N)CCN(C(=O)CN2CCOCC2)C1 C1(C(C)(C)C)C(=O)N1.c1(C(=O)OC)cc(CCC(=O)N2CC(N(C)C)C2)c[nH]1 c1(C(N2CC(NC(CCC=C=C)=O)C3(C2)CC3)=O)cnn2c1CC(C)CC2 c1(CC)cc(NC(C23CCN(C(c4cccc(C)c4)=O)CC2C3)=O)cnc1C N1(CC)CCC=C(c2ncsc2C(=O)Nc2nccc(C(=O)OC)c2C)C1 c1(C(N2CC(COC)N(C(c3ccc(Cl)[nH]3)=O)CC2)=O)cccc2c1CCO2 C1(NC(CCOC)=O)CCN(C(c2sc(C3CCCC3)nc2C)=O)CC1F c1(-c2n(Cc3ccccn3)nc(C3CCC3)n2)ccc2n[nH]cc2c1Cl.C1CCC1 c1(CC(=O)NC(C2(C(=O)NC(C(COC)C)C)CC2)C)ccc(F)nc1 c1(C(=O)NCCN(C(C)C)C(c2ccc(Cl)[nH]2)=O)ccc(NC(C)=O)cc1F Cc1cc(C(=O)NC2CCN(C(c3ccc(C4CC4)s3)=O)CC2C)c(O)nn1 N1(C(CCc2c(C)noc2)=O)CC(NC(=O)C(n2cc(Cl)cn2)C)C(C)C1 C1(N(C)C)CC12CN(C(=O)Nc1nc(-c3ccn(C)n3)cs1)C2 c1(C(=O)NCCO)ccnc(N(C2CCCCC2)C2CC2)n1 C(=O)(C1CNC(=O)c2ccccc21)N1CCC2(CN(C(CSCC#N)=O)C2)CC1 C(CCC(N)=O)(C(=O)NCC1CCC1NC(=O)CCS(=O)(=O)N(C)C)NC(C)=O C1(NC(C2ON=C(C(C)C)C2)=O)CN(C(=O)C(C)(C)O)CC2(CC2)C1 CCCCC(CC(=O)N(C)CCOCC1CC1)NC(=O)C(C)(C)N=[N+]=[N-] C1(O)(CNC(=O)C=Cc2cscn2)CCN(C(C2(c3ccccc3)CC2)=O)CC1 Cc1nc(=N)[nH]cc1C(N1C2CCC1(CNC(c1cnns1)=O)CC2)=O C1(OCCOc2nccc(C(=O)OC)c2)CN(C(c2ccon2)=O)CCC1F c1(C(N2CCC(N(CCC)C(c3cnsc3)=O)C2)=O)cc(SC)oc1C C1(C(=O)NC(C)C(C)(C)C)CCN(C(=O)C=Cc2ccccc2)CCO1 C(=O)(C1=CCCCO1)NC(C(C)(C)NC(CCc1onc(C(C)C)n1)=O)C N1(C(C2(CC)CCCC2)=O)CCCOC(CNC(=O)COC2COC2)C1 N1(C(C2(C)CCC(=O)CC2)=O)CC2CCN(C(C3CC3C(N)=O)=O)CCC2C1 N1(c2nnc(SCc3n(CC)ncn3)n2CCC(=O)OC)CCn2cccc2C1 C(=O)(C1CCc2ccccc21)NCCC(C)NC(=O)C=Cc1ccc(F)c(F)c1 N1(C(CC)=O)CCCC1C(=O)NCC(CC)NC(=O)CCSC CCC(O)(CN1CCCC1c1ccc(F)cn1)C(F)(F)F CCCCCC(C(=O)N(C)CCN(C(c1cnnc(C)c1)=O)C(C)C)C(C)C Cc1ccc(CNC(C2C=CC(NC(C3C4CCCC34)=O)C2)=O)nn1 C1(CNC(c2n(CC(=C)C)nnn2)c2csnc2OC)CCC(SC)CC1 c1(C(=O)NCC(CCNC(=O)CC2CCSC2)OC)cnc[nH]c1=N C(=O)(C(F)C(C)(F)F)NC1(C(N(CC(O)CO)C)=O)CC(CO)C1 c1(CC(C)C)c(C(N2CC(CN(C)C(C3CC3(F)F)=O)C2)=O)cnn1C CC1(C)CCOC1C(N1CCCC1(C)CCC(=O)NCCCC(N)=O)=O N1(C(c2scc(CC)c2)C(=O)NCCSC)CCOCC1C#N CCC(O)C(F)(F)C(=O)NCC1(F)CCN(C(C2CCCNS2(=O)=O)=O)CC1 CC(C)CC(C(=O)NC(C)C(C)NC(c1cnco1)=O)N(C)C C(=O)(C(F)(F)C(C)O)NCC12C(CN(C(C(C(C)C)NC(COC)=O)=O)C1)C2 C=CCC(CC)C(=O)NCC1(F)CN(C(c2nc(C(C)C)ncc2NC)=O)C1 c1(C(N(C(CC(=O)N(C(c2ccncn2)C)C)C)C)=O)sccc1C#N CCCCCS(=O)(=O)CC(=O)N(CC)CC1CCCN(C(C2SCCCS2)=O)C1 N12CCC(C1)CCC(=O)NCC2=O.CCCCCN(CC)CC.C(C)(C(=O)NC)O Cc1ncn(C)c1C(N1CCOC(CCCNC(c2ccco2)=O)C1)=O c1(C(C(=O)NC2CC(CC)C2)N(C(C(=O)OC)C2CC2(Br)Br)C)ccc(F)cc1 C1(NC(C=CCC)=O)C2CC1N(C(c1ccc(Cl)cc1OC)=O)C2C C1(NC(=O)Cn2ccc(Br)n2)COCC1NC(C12CCC1C2)=O N1(C(c2nc(CC)sc2)=O)CCN(C(=O)CC2(C)CC2(F)Cl)C2(CCC2)C1 C1(C(=O)N(C(C)C(=O)NC2CC2(C)C)C2CC2)(SC)CCC1 CCCCC(CC)CC(=O)NCC1CCC(C(=O)N(C2CCN(CC)C2)C)CC1 N1(C(c2cnc(C)nc2)=O)CCC(O)C(NC(c2cnsc2)=O)C1 CC(C)CC(C)(C)C(=O)NCCN(C1CCCCCC1)C(=O)C(C)c1ccco1 c1(NC(C2CC(F)CN(Cc3ccc(C(=O)O)o3)C2)=O)cc(F)ccc1[N+](=O)[O-] c1(CNC23CC(NC(c4ccn(C(C)C)n4)=O)(C2)C3)c(Br)cnn1C C1(F)(C(=O)NCCOCCCNC(=O)C=CBr)CC12CCCCC2 c1(C(N(C2CCN(C(C3CC4CC4C3)=O)C2)CC)=O)c(C(F)F)cnn1C C1(NC(C2(CC)CCCO2)=O)CC2CC1CN(C(=O)CC1CCOC1)C2 c1(C(=O)NC2CC(C)(NC(C3ON=C(CC)C3)=O)C2)cc(F)cc(S(N)(=O)=O)c1 c1(CNC(C2CC(O)(CC)C2)=O)cccc(NC(C2CCN(C)C2)=O)c1 N(C(=NCc1ccc(C)o1)NC(C1CCCO1)C)Cc1onc(COC)n1 Cc1cc(C(N2CC(CCNC(C3C4CC4C4CC34)=O)C2)=O)c(C)cn1 c1(C(=O)NC2CC(O)(CNC(C3(C)CC(=C)C3)=O)C2)ccccc1C(C)=O c1(NCC=CCOC(C2N(S(C)(=O)=O)CCCC2)=O)cc2ccc(Cl)cc2s1 CN1CCN(C(c2c(CNC(C3CCCC(O)C3)=O)nnn2C)=O)CC1=O C1(NC(CCCOCC=C)=O)CCN(C(c2ncccc2CO)=O)C(C)C1 c1(-c2cnc(NC(C(F)=C(C)C)=O)nc2C(N)=O)ccc2c(c1)oc(=O)n2C Cc1c(C(=O)NC2CCC2NC(=O)CS(N)(=O)=O)cncc1F c1(OC)cc(C)cnc1C(=O)NC1(C)CC(NC(C2CCOC(=O)CC2)=O)C1 C(=O)(C1=NNC(=O)C1)NC(C)(CNC(c1coc(C2CC2)n1)=O)Cn1cccn1 C1(C(CNC(c2n(CC#C)ccc2)=O)(C)O)CCN(C(c2cscc2Cl)=O)CC1 N1(C(c2c(C)n(C3CCC3)nc2)=O)CCN(C(=O)C2=CCCCO2)CC(O)C1 c1(C(=O)NC2CCC(CCNC(C3(C)CC(F)(F)C3)=O)C2)ccc2ccnn2c1 S(=O)(=O)(c1c(OC(F)(F)F)ccc(Br)c1F)NCC1C(C)OCC1 CC1(C)CCCN(C(=O)CCC2CCC2)C1C(N1CCC(OCCF)C1)=O c1(NC(C(CCOC)NC(COCCC)=O)=O)ccc(C)c(O)c1C C1(CNC(=O)CCC2CCC2)CCC(CNC(C23CC(CO2)C3)=O)CC1 N1(C(C(=O)NCCC)C(C)C2CCCCC2)CCCCC2(CCC2)C1 Cc1ccc(NC(=O)CN2C(CO)COCC2C)cc1Cl c1(C(C(N2CCC(NC(C(C(C)C)OC)=O)C2)=O)C)cc2ccccc2o1 C12(NC(=O)C3=CCCOC3)CCN(C(=O)COc3cn[nH]c3)CCC1C2 C=CC1CN(C(c2csc(C3CCCCC3)c2)=O)CC1NC(=O)C#CC1CC1 C1(CC(N2CC(C(Cn3cc(COC)nn3)F)C2)=O)CC2(CCCC2)CO1 N1(C(c2ccc(O)nc2)=O)CCC2(CCC(N3CCCCCC3)CC2)CC1 N1(C(c2cc(C)c(C)o2)=O)CCN(C(=O)C(C)CN(C)C)CC1C1CCC1 C12(CC(=O)NC3CC3NC(=O)C(C3CCOCC3)O)CCC(CC1)OC2 c1(OC)cc(N)c(C(=O)NC(C)C(C)NC(c2cc(Cl)sc2Cl)=O)cc1F c1(NC(C2C(NCc3ccc(C(=O)OCC)[nH]3)C2)=O)ncc(Br)nn1 c1(C(C)C)ccc(NC(C2(CF)CN(C(=O)C(C)OC3CCCC3)C2)=O)s1 c1(C(C2CCCCC2)O)ccccc1OCC(F)F.c1(CC)nnnn1C1CC1 C1(C)(OC)CC2CC1CC2NC(=O)NC(c1ccc(N2CCCCC2)cc1)C N1(C(C(Cc2cn[nH]c2)NC(c2c(CC)cns2)=O)=O)CCN2CCCCC2C1 C(=O)(C(C(C)(C)C)NC(C)=O)NCC(CC)(CC)NC(C(C)OCCCC)=O c1(C(=O)NC(C(=O)NC2(C#C)CCOC2)(C)CO)ncc2ccccn12 c1(CC(C(=O)N(CCCNC(=O)C(C)O)CC)C)ccc(OC(F)F)cc1 S(=O)(=O)(C1CC1)NCC(=O)NC(C1CCN(C(C2CCC2)=O)C1)(C)C CC(C)CC(C)(CNC(=O)CCc1ccsc1Cl)NC(C1CCOC1)=O N1(C(c2n(COC)ncc2)=O)CCOC(CNC(=O)C(O)C2CCC2)C1 C(=O)(C(C(C)(C)C)N(C)C)NCC(CC(=O)NC(Cn1ncc(C)c1)C)O c1(CC(=O)NC(CN(CCC(=C)C)C)C)c(Cl)cccc1Cl N1(C(c2c(CC)cccn2)=O)CCC(NC(=O)Cc2cc(C)[nH]n2)C(C)C1 N1(C(c2cc(OC)no2)=O)CCN(C2CN(C(C3CCCC3(F)F)=O)C2)CC1 c1(N(CCC(N)=O)C)nc2cc[nH]c2c(=NC2CCCn3ccnc32)[nH]1 C1(N(C(c2c(F)ccc(COC)c2)=O)C2CC2)(CO)CC2(CCOCC2)C1 C12(CNC(c3cc(C(C)=O)sc3)=O)CC(C1)C(NC(=O)CCC(C)(C)C)CO2 C(=O)(CS(=O)C(F)(F)F)NCC1CC(NC(c2cn(C)nc2O)=O)C1 N1(C(c2c(C(=O)OC)c[nH]n2)=O)CC2CCC(C1)C2NC(c1cc(Cl)ns1)=O c1(OC)cc(N)c(C(N2CCC2CC(=O)NC2CC(OC)C2)=O)cc1Br CCC(C)(O)C(=O)NCC(C)(O)CNC(=O)CC(=O)OC(C)(C)C CCCCC(C(=O)NCC1CCCC1NC(c1cc(Cl)no1)=O)NC(N)=O Cc1nn(C)c2ncc(C(N3CCC(OC)C3)C(=O)NCc3ccccc3)cc12 C1(CNC(CCOCC#C)=O)CN(C(=O)CSc2nnnn2C)CC12CCC2 c1(C(N2CCCC(C(C)(C)O)C2)C(=O)Nc2c(C)cccc2)ncc(Br)cc1C c1(C2(C)CC2)ccc(C(=O)NCC2CCCCN2C(=O)CC2CC(CF)C2)cc1 N1(C(C2C(CC)CCCC2)=O)CC2(CO)CC1(C(=O)N(C)Cc1ncco1)C2 N=c1[nH]c2cc(C(N3CC(C(N)=O)(CNC(=O)CC4CCC(O)C4)C3)=O)ccc2s1 C1(F)(CC)CCN(Cc2cccnc2O)CC1 C1(COC)(CNC(=O)CN2CCCC2C)CN(C(=O)CCc2cnn(C)c2)C1 C(=O)(C1=C(Cl)CC1)NC(CNC(=O)CCc1ccc(Cl)s1)CO c1(C(N2CC(C(N3CCC(N(C)C)C3)=O)NCC2)=O)ccc2scnc2c1 C1(NC2(c3nnnn3C3CCCC3)CC(C(F)(F)F)C2)CCCCC1CO CC1(O)COCCN(C(C2COCCC2NC(c2cc(F)cc(F)c2)=O)=O)C1 c1(C(N(CC(COC(C(=O)OC)CSC)(C)C)C)=O)ccc(Cl)cc1Br c1(CNC2C(C(=O)Nc3onc(C)c3Br)C2)ccc(Cl)c(F)c1 N1(C(C(F)=CCC)=O)CC2(C1)CN(C(c1cnc3[nH]c(O)nc3c1)=O)CCO2 S(=O)(=O)(c1cccc(C(=O)NC2(CN(C(=O)CN(C)C)C)CC2)c1)N(CC=C)C C(C(O)CN=c1ncnc2[nH][nH]c(C)c1-2)NC(C(CCC)OCC)=O c1(OC)ncc(Cl)c(=NCC2CC(C)N(C(c3cc4n(n3)C(C)CCC4)=O)C2)[nH]1 N1(c2cc(NC(c3cccnc3N(C)CCO)C)ncn2)CCN(C)C(CO)C1 N1(C(=O)C2=COCC2)CC2CC1CCN2C(C1COc2ccccc2C1)=O c1(C(N2C(C)CN(C(=O)CCOCC(F)(F)F)CC2)=O)cnn2ccc(O)nc12 N1(CC)CC(C)N(CCN2CCC(n3cnc(C(=O)OC)c3N)CC2)CC1C CCCCCC(C(=O)NC1(C)CCN(CCCSC)CC1)NC(S(=O)(=O)CC)=O C1(C(NOCC=C)=O)CCN(C(c2cnncc2O)=O)C1C(C)C CCCC(C(=O)N1CCN(C(=O)Cc2cncnc2)C(CO)C1)C(C)C c1(C(=O)NC2(C)CN(C(C3COC(=O)O3)=O)C2)cccc(C(F)(F)F)c1N c1(CC)c(C(N2CCCCC2c2cn[nH]c2)C(=O)NCCC#N)cccc1C Cc1cc(Cl)cc(C)c1C(=O)NC1CCCN(C(C2CCNC2=O)=O)C1 CC(C)C(C(=O)N)Oc1ccccc1Br.C(CCCCSCC)NC(=O)CN C(CC(C)C(=O)NCCCCNC(C1CC(O)CN1C(C)=O)=O)OC c1(C)ccc([N+](=O)[O-])o1.c1(C2CCNC2)ccc(I)cc1.C12C=CCN1C2=O c1(OC)c(C)cnc(CCNC2CCc3ccccc3C2)c1C c1(C(=O)NC(C(C)NC(=O)Cn2nnc(=O)[nH]2)CO)ccc2c(c1)OCC2 N1(C(C(CC2CN(C(C(N3CCOCC3)C)=O)C2)F)=O)CC(C2CCCCC2)C1 C1(CC=C)(C(=O)NC2COCC2C=C)CCCN1C(C12CC(F)(C1)C2)=O c1(C(N2CC(CNC(CC(C=C)C)=O)OCCC2)=O)ccc2nsnc2c1 N1(CCNCc2cc(CC(=O)N(CCC)CCC)no2)CCC2(C1)OCCO2 O=S1(=O)CCC(C(c2nnnn2C2CCCC2)Nc2cnc(C3CC3)cn2)CC1 Cc1ccccc1CS(=O)(=O)NC(c1c[nH]nc1C(F)(F)F)=O Cn1cccc(C(N2CCC(O)(CNC(=O)C(c3ccc(Cl)cc3)O)C2)=O)c1=O C1(CNC(CCOCCC)=O)Cc2ccccc2CN1C(=O)C(C)OCCOC c1(C(=O)NC2(C)CCN(C(c3ncc(CC)nc3)=O)C2)ccc2scc(C)c2c1 CN1CCN(C)CC(NC(=O)CCC2(C)CN(C(=O)CC3(O)CCC3)C2)C1 N1(C(c2c(C)scn2)=O)CC2(CCCC2N=c2ccnc(S(C)(=O)=O)[nH]2)C1 C(=O)(C(CCOCCO)NC(=O)C=CCO)NC(C)Cc1nn[nH]n1 N1(C(c2cc(C(C)=O)[nH]n2)=O)Cc2ccnn2CC(NC(=O)C(O)CN(C)C)C1 c1(C(=O)NCC2C(NC(=O)CN3CC=CC3)C2)cc([N+](=O)[O-])c[nH]1 CC(C)C(C)(CNC(c1cc[nH]c1)=O)NC(=O)C(C)n1ccnc1 CCCC(C(O)C(=O)N1CC(=O)NCC1CC)NC(=O)C(O)C(F)(F)F Cc1ccnnc1C(=O)NCC1(C)CCN(C(c2ccc(F)s2)=O)C1 CCCCC(CCCC)NC(C1(C)C=CCN1C(C1OCCC1C)=O)=O CCCC(CC)CC(=O)NC1(CNC(=O)C(C)CSC)CC1 c1(C(=O)NCC(CC=C)NC(C2CSCC(=O)N2)=O)cnc(C)cc1C C1(N(C(C(C=C=C)C)=O)C)CCN(C(=O)Cc2ccc(O)cc2Cl)CC12CC2 O=C1CCC(CNC(=O)N(C2CCCC2)Cc2ccccc2Br)CN1 N1(C(C2(COC)CCOC2)=O)CCC(CNC(c2c[nH]nc2)=O)CC1.C(C)(=O)O Cc1oc(CO)cc1C(=O)NCC(C)(O)CNC(=O)Cn1cccn1 N1(CC(=O)NC(CNC(C)=O)(C)C)CC(C(F)(F)F)CCC1C(F)(F)F C#Cc1cc(F)c(C(=O)NC2(CC=C)CCN(C(C3CC(C)=NO3)=O)C2)cc1F Cc1cc(N2CCC3NCCC3C2)nc(=NCc2nc(C(F)(F)F)cs2)[nH]1 C1(F)(CNC(C(C)NS(CC)(=O)=O)=O)CCCN(C(c2cc(Cl)c(C)cn2)=O)C1 c1(C(=O)NC(C(CO)NC(C(CC)n2cccn2)=O)C)ccnc2c1cnn2C N1(C(c2cc(C)sc2)=O)CCC2(CC1)CC(CNC(=O)CSc1cnn(C)c1)C2 c1(CNC(N2CCN(c3c(Br)ccc(C)c3)CC2)=O)c(C)cc(Br)cc1F C#Cc1cnn(C)c1C(=O)NCCCCCCN(C(=O)Cc1ccnn1C)C Cc1ccc2c(c1)CC(C(N1CC3C(NC(=O)CC(F)F)C3C1)=O)S2(=O)=O CCCCCC(O)C(=O)NC1C=CCN(C(c2cc(Br)cc(F)c2O)=O)C1 C(=O)(C(C)(F)C(F)(F)F)NCCCC(C)NC(c1c(C)[nH]c(C)c1C)=O C1(NC(c2c(C)nc(C)[nH]2)=O)CN(C(=O)Cc2ccnn2C2CCC2)CCC1F C#Cc1ccc(C(=O)NCCC2CC(F)(F)CN2C(c2occc2CC)=O)cc1 C(C(F)(C(=O)NCc1ccc(CO)o1)C(C)C)NC(c1[nH]cc(C)c1C)=O C(CC(C(N)=O)NC(=O)C(C1(O)CCCCC1)NC(=O)CCOCC1CC1)OC CC(CCC(=O)NCCC1CCN(C)CC1)NC(c1cc(C2CC2)no1)=O C12(C(N3CC4C(CC(=O)NC(C5CCOC5)C#C)C4C3)=O)CCCC1C2(F)F CN1CCN(CCC(=O)NCC(C2CC2)NC(=O)Cc2nccn2C)CC1 C12(C(=O)NC(CC)C3CC3)CCC(NC(C3CCOCC3(C)C)=O)(CC1)C2 Cc1c(CNC(=O)C(=O)NCc2ccnc(Br)c2F)cccc1F C1(CNC(C(=O)NCc2ccc(N3CCCNC3=O)cc2)=O)CC(O)C12CCC2 Cn1nnc(CNC(c2ccnnc2)=O)c1C(N1CCCC(CF)C1)=O c1(CC(=O)N(CC(C)CNC(c2cn(C)nc2O)=O)C)ccc2c(c1)CCOC2 n1(CC(=O)NCC2CCN(C(c3cc(C)c(Cl)s3)=O)C2)cccc(N)c1=O c1(C(NOC(C(=O)N2C(C(CC)OC)CCC2)CC)=O)cc(C#N)c[nH]1 N1(C(C(N2CC(C)C2)C)=O)CC(CC(=O)NCCN(CC(F)F)C)C2(CC2)C1 c1(C(=O)NC2(C)CN(C(=O)CC3CCOC(C)(C)C3)C2)nn2c(c1Br)CCC2 c1(COC(c2ccc(C(=O)OC)o2)=O)c(C)cc(Cl)cc1C N1(C(c2nc(CC)oc2)=O)CC2CN(C(C34CCCC3C4(F)F)=O)CC(C1)O2 CCC(C(=O)NCC)N(C(Cc1ccco1)C(=O)N1CCC(CC)C1)CC1CCC1 c1(C(=O)NC(CN(C(c2cnc(C(C)C)o2)=O)CC)C)cnn(C(F)F)c1 N1(c2cc(N(CCOCCC)C)nc(COC)n2)CCCC(C2CCC2)C1 C1(NC(CC2CC(=C)C2)=O)CN(C(=O)CCN(C)C(C)=O)C2(CCCCCC2)C1 N#Cc1c[nH]c(C(=O)N(C2CC2)CC2CCCN2C(c2ccc(C(N)=O)[nH]2)=O)c1 C(=O)(CCCC(CC)NC(c1cnnc(O)c1)=O)NCC(C)OCC=C N1(C(CC2C(CC)CC2)=O)CC(CNC(C2(CO)CC(OC)C2)=O)C(C)(C)C1 CC1=NC(C)(CNc2cccc(C(C)NC3CCNCC3)c2)CS1 C12(CNC(C(COC)(C)C)=O)CCC1CCN2C(=O)CCCc1nc(C)no1 C(=O)(CCC(C)CCCC)N(C1CCCCCC1)CCNC(C(C=C)CC)=O C(c1ccc(Br)o1)=C(C)CC(=O)CS(=O)Cc1nc(-c2ccsc2)no1 c1(C(C)C)ccc(C(=O)Nc2ccc(CCO)cc2)cc1.N12CC(C)CC1C2=O c1(C(N2CCCC(NC(C3ON=C(CC)C3)=O)C2)=O)cccc2c1CCCN2 N1(C(C2CN(C)CC2C(F)(F)F)=O)CCCC2CN(C(=O)C(F)(F)C3CC3)CC12 c1(C(N(CC(C)NC(=O)COCCCOC)CC)=O)cc2ccccc2cn1 C12(CNC(C#CC(C)C)=O)CCCC1N(C(=O)Cc1nc[nH]n1)CCC2 C1(CC)CCCC1C(N1CC(N(C)C(c2cnn(C3CCOCC3)c2)=O)C1)=O CC1=NOC(C(=O)NC(C)CCCNC(=O)C=CCO)C1 N1(C(c2n(CC=C)ccn2)=O)CC(NC(=O)Cn2cc(C(=O)OC)cn2)C(C)C1 CS(=O)(=O)c1ccc(C(=O)NCC2CCC2NC(=O)Cc2cccnc2Cl)[nH]1 C1(NC(c2c(CC)cno2)=O)CN(C(C2CCN(CC(C)C)C2)=O)CC1C(F)F c1(C(=O)NCC(C2CCCCC2)NC(C2C(C)C2C)=O)cnc2nccn2c1 n1(CC)cc(C(N2CCCC(CN(C)C(C3CC3(F)F)=O)C2)=O)c(C(C)C)n1 CC1CC(NC(c2coc(C3CC3)n2)=O)CCN1C(C12CCC(C1)OC2)=O C(=O)(C#CC(C)(C)CNC(c1oc(CO)cc1C)=O)NCC(C1CCCC1)OC N1(C(C2C(=C)C2)=O)CCC(CNC(=O)C=Cc2cscn2)C(O)C1 C(=O)(C1Cc2ccccc21)NC(CC=C)C(N1CC(C)C(C)(CO)C1)=O C(c1cnc(O)nc1O)=CC(=O)NC1CCCN(C(=O)CCCc2cncs2)C1 C1(C(N2CC(O)(CNC(Cn3ccc(C)n3)=O)C2)=O)CCN(C2CC2)C1=O Cc1cccnc1CC(N1CCC(CN(C(=O)CN2CC(C)(C)C2)C)C1)=O CC1(C)CC(CNC(=O)C(C2CCC2)NC(C23CC(F)(C2)C3)=O)CO1 c1(C(=O)NCC2CN(C(COC(CC)C)=O)C(C)C2)cccc(N=[N+]=[N-])c1 Cc1ccc([N+](=O)[O-])c(C(=O)NC(C)CN(C)C(c2cc(Cl)c(Cl)cc2N)=O)c1 C1(NC(C(C=C)c2ccccc2)=O)CCCCN(C(=O)C(C)C2CC2)C1 c1(C(=O)NCCC(C)NC(=O)C(CN2CCCC2)c2ccccc2)ccc(Cl)o1 C(C1=CCCN(C(C2C3CCC(=O)C23)=O)C1)NC(CC1(C)CC1)=O Cc1cnc(C(=O)OC2CCN(C(=O)OC(C)(C)C)CC2F)cc1C CN=c1[nH]c(C(=O)NCC2CC(F)CN2C(=O)CCC(F)F)cs1 C(=O)(CC(C(F)(F)F)NC(=O)CC1CCCC(=O)N1)N1CC(C)(C)C1 c1(C(=O)OC)ccc(F)c2c1CN(Cc1nc3ccccc3n1CCOC)C2 c1(C(=O)NC(C)CCNC(C2CC(=O)CO2)=O)ccc(Cl)cn1 CN=c1ccc(C(N2CC3(CC3)CC2C(=O)NCCC2CC2C)=O)c[nH]1 c1(C(=O)NCC(C(C)C)NC(C(C)OC)=O)cccc(OC(C)C)c1 C1(CC)C(NC(c2sccc2C)=O)CCCN1C(C1(F)CCOC1)=O N1(c2n(CCOCC=C)c(C3(C)CCOC3=C)nn2)CC2OC(C)(C)OC2C1 C1(NC(C(c2ccccc2Cl)(C)C)=O)CN(C(C2CC=CCC2)=O)CC1O C1(c2c(C)ncs2)CCN(C(c2cccc(Br)n2)C(=O)NC2CCC2)CC1 N1(C(C(C)OCC)=O)C(C(=O)NCC(C)(C)CCOC)CCC1C C1(C(=O)NCCC2CCCN(C(C(CC)n3cncn3)=O)C2)CCC2(CC1)N=N2 CCC(CC(=O)NC1CN(C(c2cccc[n+]2[O-])=O)C2(CCC2)C1)C(C)(C)C CC1CC(NC(=O)CCCc2ccc(F)cc2)CN1C(C12CCC(C1)C2)=O C(C(C)(C)CNC(C1(C)CCCC1)=O)C1CN(C(CSCC=C)=O)C1 C#CC1CN(C(C2CCCC2NC(c2[nH]cc(C)c2C)=O)=O)CC1O c1(OC)c(CN2CCC2C(=O)NCC(O)CCO)cccc1F N1(CC)CCN(CCC(=O)NC(CNC(=O)C(C(C)C)OC)CO)CC1 N1(C(C(CCF)NC(Cn2c(C)ccn2)=O)=O)CCC2(C=CCO2)CC1 c1(CNC(=O)CC23CCCC2C3)ccc(OCC(F)(F)F)nc1.CCO C1(C(N(C)Cc2n(CC)ccn2)=O)CC(NC(=O)C=CC2CCCC2)C12CCC2 c1(-c2cccc(CC)c2)cccc2[nH]nc(C(=O)NC3CCCOC3)c12 c1(C(N2C(C)CCC(NC(c3occ(C(N)=O)c3)=O)C2)=O)c(F)cc(N)cc1F N1(Cc2n(CC)cnc2)CCC2(CC1)CC2(C)C(=O)N(CC(N1CCCC1)=O)C C(=O)(C1=C(Cl)CCCC1)NCc1nccc(C(N2C(CC)CC(O)C2)=O)c1 c1(N2CCC(OCCNC(CC(C=C)c3ccccc3)=O)C2)ncnc(Cl)c1Br C1(OC)CC(C(=O)NC(C)(CNC(=O)CCn2ccccc2=O)CO)CC1OC C1(NC(c2c(C)cco2)=O)CCC(C)N(C(c2ncc(Cl)cc2F)=O)C1 Cc1[nH]nc(C(N2CCCC(CN(C)C(C3CC3F)=O)C2)=O)c1Br Cn1nc(CNC(=O)CN(C2CCC2)C)cc1C(=O)NCC(O)C(N)=O Cc1cc(C(=O)N(C)CC2(O)CN(C(=O)C(F)(F)CC3CC3)C2)c(N)c(Cl)n1 c1(C(=O)NC2CC(CNC(=O)C(C3CCCCC3)F)C2)cccc(O)n1 C1(C(=O)NC(C)CC2CN(C(=O)Cc3cscn3)C2)CCn2nccc2C1 C(=O)(C(CCF)NC(=O)CP(C)(C)=O)NCCC1(C)OCCO1 c1(C(N2CC(NC(C(CC)SC)=O)C(O)CC2)=O)ccc2cnccc2n1 Cc1cc(C(=O)NC2CC(NC(=O)CCc3ccc(F)cc3Cl)C2)cc(C)n1 N1(C(C(CCC)C)=O)CC(C)(CNC(c2c(Cl)cnn2C)=O)CC1(C)C CCCCCCCC(C)NC(=O)C#CCNC(=O)CC(C)=C(C)C Cc1ccc(C(N2CCCN(C(c3ncsc3C3CC3)=O)CC2C)=O)c(N)c1C C(C(=O)C1CCCc2ccccc21)OC(CN=c1ccc(C#N)c[nH]1)=O c1(C(N2CCN(C(C3C(=C)CC3)=O)C(C3CC3)C2)=O)cc(C)c(F)cc1Cl C1(C(=O)O)C(O)CCCN1C(c1ccc(-c2ccc(C3CC3)cc2)cc1F)=O C1(OC)CCC(C(=O)NC2(CCNC(=O)COCc3nccn3C)CCC2)CC1 C1(NC(Cn2c(C)cnc2)=O)CCCN(C(=O)CCc2ccc(Cl)nc2)C1C Cc1ccc(OCCC(=O)NCC(C)NC(c2nccnc2N)=O)c(Br)c1 N1(C(C2(C)CCC(=O)NC2)=O)CC2CN(C(C3CC(=O)C3C(C)(C)C)=O)CC2C1 C(C(CNC(C1(c2n[nH]cc2C)CC1)=O)C(F)(F)F)NC(C=C(COC)C)=O CCCCC(O)CC(=O)N(CC(C)NC(c1cnc(OCCOC)c(Cl)c1)=O)C C1(C(=O)NCC(C)CN(C(=O)CC2OCCO2)C)CCC(F)(F)CO1 C#Cc1cncc(C(=O)NC(CC(=C)Cl)C(=O)N2CC(c3ncccn3)C2)c1 c1(OCC)cccnc1C(N1CCC(C2CCCN2C(C2CCCN2C)=O)C1)=O N1(C(C(C)Br)=O)CC2(CCC(CNC(=O)C(Br)Cc3ccccc3)O2)C1 CCCCCCCCNC(=O)CNC1CN(C(c2ncn(C(C)C)n2)=O)CC1F CC1CC(NC(c2nc(Cl)nc3c2CCC3)=O)CC(C)S1(=O)=O c1(C(=O)NCCCN(C(C(C)OCC)=O)CC)cncc(NC)c1 c1(OC)ncnc(N2C(C(=O)Nc3ncc(F)cc3Br)CC3CC23)c1C N1(C(c2cc(C3CC3)nn2C)C(=O)NCCCCCC)CCC(O)C(F)(F)CC1 N1(C(CC2N(C)CCC2)=O)CCSCC1C(=O)N(CC(c1nn[nH]n1)C)C N1(C(=O)Cn2cccn2)CCC2CCN(C(=O)C=C(Cl)Cl)CC2C1 c1(CN2C(C(=O)Nc3ccc(C(=O)OC)nc3)CC(C)C2)cccc(C)c1O C1(CNC(C2C(C(=O)OC)COC2)=O)CC(C)CCN1C(c1ccnc(C)n1)=O c1(C(=O)NCC(CN(C(=O)C(F)=C2CCCC2)C)O)cccc(C2CC2)n1 c1(C(=O)NCCN(C)C(C2CCC2F)=O)ccc2c(c1)CCNC2=O N1(C(C(C)OCC=C)=O)CC(n2cc(-c3ccncc3Cl)nn2)C(C)C1 C1(C(=O)NC(COC)C(C)C)CCN(C(=O)CN2CCNC(=O)C2)CC1(C)C CCCCCC(O)C(=O)NC1CN(C(=O)Cc2sc(C3CCC3)nc2C)CC1C Cn1[nH]c(=NC(=O)CSc2c(F)ccc(F)c2Br)cc1C1CC1 CC(F)(F)CCC(=O)NCc1cc(C(=O)NCCCC(O)CO)n[nH]1 C1(NC(CCc2c(C)n(C)nc2)=O)CCN(C(c2cccnc2S)=O)CC1O Cc1cnc(C(N2CCC(NC(c3cn(C4CCC4)nn3)=O)C(O)C2)=O)c(C)c1 c1(CCC(N2CCC(C(C)NC(c3c(C)con3)=O)CC2)=O)nnc(O)nc1O C1(NC(C#C)=O)CC2(C1)CN(Cc1cc(Br)cc(I)c1)C2 CC1CCC(C(N2CCC(CN(C)Cc3ncoc3C3CC3)C2)=O)CC1 N1(C(Cc2c(C)occ2)=O)CC2CCN(C(=O)CC3(C)CCCO3)C2C1 Cc1cc(C(=O)NCC(F)CNC(=O)CCC(=O)c2cccs2)[nH]c1C C1(NC(CN(C2CCC2)C)=O)CCN(C(=O)COc2ccc(F)cc2)CC1(C)C C=CCC(C)(CC)C(=O)NCC1CCCN1C(=O)Cn1cccc(C)c1=O Cc1c([N+](=O)[O-])ccc(N2CC(c3cc(F)cc(F)c3)(O)C2)c1I C1(C(=O)OC)C(OC)C(OC)CN1Cc1sc(C)c(C)c1Br c1(C(C)NC(c2n(CCC)nnn2)C=Cc2ccccc2)ccc(C#N)cc1 c1(OC)cccc(CC(=O)C(=O)NC2CC(CNC(c3cnc(C)[nH]3)=O)C2)c1 N1(CCCNC(c2cnc(OCC)s2)=O)CCN(C(c2nc(Cl)sc2C)=O)CC1 N1(C(CNC(C(CC)C)=O)=O)C(C(=O)NCc2[nH]c(C)nc2C)CCC12CC2 c1(CC)oc(C)cc1C(=O)NCCC(C)(C)NC(C1(OC)CCCCC1)=O c1(C(C(=O)N(CCCOCCNC(c2cnco2)=O)C)(F)F)ccc(F)cc1F c1(OCCCN(C(=O)C=Cc2ccc(F)cc2)C)ccc(Cl)cc1Cl C1(C)(C(=O)NC2C(SC)CN(C(c3cc(O)cs3)=O)C2)CCCC1(F)F CC1(C)CC(=O)N(CC(N2CC=CC(NC(=O)Cc3ccnc(Cl)c3F)C2)=O)O1 C1(NC(CC(CCC)C)=O)CCCC12CN(C(c1cc(O)ccc1O)=O)C2 C(CC(=O)NCCCCCO)(C(F)F)NC(C(CC)=CC)=O C(=O)(C#CC1(C)CC1)NCC(CCCC)NC(=O)C(C)Cc1cccnc1 CC(C)C(C)CC(=O)NCC(CC1CC1)C(=O)NC1(c2nc[nH]n2)CC1 Cc1cncc(C(=O)NC(CNC(=O)C(=O)N(C)C)C(C)(C)C)n1 C1(Cn2cc(C(CC)O)nn2)CCN(C(c2ccnnc2O)=O)CC1(F)F c1(C(N(C=O)Cc2cc(Br)c(F)cc2F)C)ccc2c(c1)OCCO2 Cc1oc(-c2ccco2)nc1CC(=O)Nc1cncc(OC(C)C)c1.C(=O)C(C)C N1(C(CCSC)=O)CC2(CCC(CNC(C3CC3CC(C)(C)C)=O)O2)C1 C(=O)(CCC1=NNC(=O)CC1)N1CC(O)(CNC(CCc2cc(OC)no2)=O)C1 C1(C(=O)NCCN(C(C2N(C)C(=O)OC2)=O)C2CC2)CCC2(CC1)COCCO2 c1(SC)ccc(C(=O)NC2(C)CN(C(=O)CC3CC(C)=NO3)C2)s1 N1(C(c2noc(C)c2C)=O)CCC2(CC1)CC2C(=O)Nc1ccc(O)cc1Br c1(C(=O)NC2C(NC(C3(C#N)CC34CCC4)=O)COC2)cnc2[nH]ncc2c1 C1(C(=O)NC2C=CC(C(=O)NC3(C=C)CCC3)C2)CC2CCC1CC2 C1(C)(OC)CCCN(C(c2cc(Cl)ncc2Br)C(=O)NC2CC2)CC1 c1(C(N2CC3C(CNC(C4CCN(C(C)=O)C4)=O)(C3)C2)=O)cccc(=S)n1O C#CC1(NC(C2C(CNC(C3CCCCS3)=O)C2(C)C)=O)CCCCC1 CC(C)(O)C(C(=O)N1CCC(c2ccco2)C1)NC(=O)CCOC1CC1 Cc1noc(C)c1CC(C)C(=O)NCC1CC1NC(c1csc(C(F)F)n1)=O C1(NC(CC=C)=O)CS(=O)(=O)CC1NC(c1nn(C(C)C)cc1Br)=O C=C(C)C1OCCC1CNC(=O)CC(C)(C)N(C)C(c1ccc(Cl)o1)=O Cc1nn(C)c(C)c1CCC(=O)NC1(CC(=O)N(CC2CC2)CC2CC2)CC1 C1(CNC(c2c(COC)ccs2)=O)CN(C)CCN1C(C1CCOC1C)=O c1(OCC)nc(Cl)ccc1NC(c1c(C)[nH]c(C(=O)Nc2cnns2)c1C)=O N1(C(C)=O)CCC2(COC(CNC(c3cc(C(F)F)[nH]n3)=O)C2)C1 c1(CNC(C(C)O)=O)cn(CCNC2(CO)CC2C(F)(F)F)nn1 c1(C(N(C)CC2CCCN(c3nc(C4CC4)ns3)C2)=O)cnc2c(Cl)cccn12 C(C(COC)C(=O)NC(C(N1CCC(COC)C1)=O)c1ccoc1)OC c1(C(N2C(CNC(C3(F)CC=CC3)=O)CC3CC23)=O)cncc2c1CCC2 Cc1nc2oc1C(=O)NC2.C1(C(C)NC(=O)CCc2nccs2)CC2(CCC2)C1 C1(C(=O)NCC#CC2CC2)(CC)CCN(C(c2cnsc2)=O)CC1 c1(NC(CCCC)CCC)ccc(S(=O)(=O)NCCS(=O)CC(F)(F)F)cc1F O=C(CCCCCCCO)N1CC2(CCC(C(N3CC(O)C(F)C3)=O)O2)C1 C(=O)(C(C)(C)C(C)(F)F)NCC1CC(OC)CN1C(C1CCCS1)=O C(=O)(C1=NOC2COCC12)NC(CCCC)CNC(c1occc1C(C)C)=O c1(OC(C(=O)NC(CCNC(C(C)=C2CCCC2)=O)C)C)cc(Cl)cc(Cl)c1 c1(C(=O)NC2C=CC(CNC(C)=O)C2)ccc2c(c1)CC(=O)N2 C1(C(=O)Nc2cccc(O)n2)CN(C(C2CC=CCC2)=O)CC(F)(F)C1 C1(S(C)(=O)=O)(C(N2CC3CC(CNC(c4nc(C)[nH]n4)=O)C3C2)=O)CCOCC1 c1(C(=O)NC(C(C)C)CNC(=O)C(C)Cc2ccco2)cc2cccnc2[nH]1 C1(NC(C(=O)N(CCCn2ccnc2)C)=O)COCC1N1CCOCC1 C1(CNS(=O)(=O)CCCl)CC2(C1)CN(Cc1c(Cl)ccnc1Br)C2 N1(C(c2cc(COC)oc2C)=O)CC(OC)C(OC)C1CNC(=O)CCC(C)C C1(CNC(C)COC2CCCCO2)Cc2cc(F)ccc2NC1=O c1(C(=O)NC2C(NC(C34CC(CCC)(C3)C4)=O)CC2)cnccc1N(C)C C1(CCC)CN(C(C2CC3(CC3)C2)=O)CC1C(=O)N(C)Cc1cncnc1 c1(C(N2CC(CNC(=O)CC3NC(=O)NC3=O)OCC2)=O)cc(Cl)nnc1O N1(C(c2cc(OC)cc(OC)c2)=O)CC(C)OC(C)(c2nnc(C)o2)C1 c1(C(N2C(CC(=O)Nc3nccc(OCC)c3)CCC2)=O)cc(Cl)cc(Br)c1 C(=O)(C(C)CN(C(=O)CONC(=O)C1CC(OC)C1)C)OC c1(CN2CC(NC(Cc3cccc(OC)c3)=O)C(O)C2)ccccc1C#N Cc1n[nH]c(C)c1CNC(=O)CNCCNC(=O)C(C)(C)C CCCC(C(=O)NCC(C(C)C)NC(c1cc(C(=O)O)n(CC)n1)=O)N(C)C N1(C(C(C)SCC)=O)CC(C(=O)NC2CC=C(C)CC2)C(C)(C)C1 N1(C(C(CC(C)C)NC(c2ncc(C)nc2)=O)=O)CCC2(CCOC2)C1 c1(-c2c(C)cc(C)s2)ccc2c(c1)CCN(Cc1cc(Br)cc([N+](=O)[O-])c1Cl)C2 c1(NC(=O)CC2CCCN2Cc2cc3ccncc3[nH]2)cccc(S(=O)(=O)O)c1 C1(C(=O)NC(=O)C(F)(F)F)CN(CC2C3CC2C(C)N3)CCC1c1ccccc1 C1(C2CN(C(=O)NC3CCC4CCC34)C2)CCCCN1C(=O)OCc1ccccc1 c1(SC)cc(C(N2CC(CNC(c3n[nH]c(C)c3Cl)=O)C3CC23)=O)oc1C C#CC1(C(=O)NCCCc2cccnc2)CN(C(C2(C)CCCC2)=O)C1 c1(C2(C(=O)NCC3(n4cc(CN5CCOC5=O)nn4)CC3)CC2)cc(Cl)ccc1F N1(C(C2(CCOC)CCC2)=O)CCC(NC(C2CCS(=O)CC2)=O)C(F)C1 Cc1nn(C)cc1C(=O)NC1(CNC(C23CC2C3)=O)CC1 c1(C(=O)NCCN(C(CC2C(C)C2)=O)C)ccc(-c2cnnn2C)cc1 c1(C(=O)NCC2OCCC(NC(C(C(C)O)N(C)C)=O)C2)cccc2[nH]ncc12 N1(C(c2ccc(C#N)s2)=O)CC2CC1CC2N1CCC1CO n1(CC)cnc2c(NC3CCC(SC)C3)[nH]c(=NC3CCCn4ncnc43)nc12 C#Cc1ccc(CC(N2CC(C(N3CC(N(C)C)C3)=O)C(COC)C2)=O)cc1 C1(C(=O)NC2C(NC(=O)Cc3cccnc3Cl)CCCC2)CC2(C1)CC(O)C2 N1(C(c2cnc(CC(C)C)[nH]2)=O)CCC2C(C1)CN2C(=O)C=Cc1cn(C)cn1 N1(C(c2c(C)c[nH]n2)=O)CC(CNC(C2CCN(C)C2=O)=O)OC(C)(C)C1 N1(C(C=C(CC)CC)=O)CC(C2CCCN(C(=O)C(CN(C)C)N(C)C)C2)C1 Cc1cc(N)cc(C(N2CCCCC2CCNC(=O)C2=CCS(=O)(=O)C2)=O)c1F C(=O)(CCCC(=O)N1CC(N(C)C(c2cc[n+]([O-])cc2)=O)C2(CC2)C1)NCCC CS(=O)(=O)C1CN(C(=O)C(N)Cc2ccco2)C2(CCOCC2)C1 c1(C(C)C)nc(NCC2CC23CC3)cc(=NC2CCn3nnnc3C2)[nH]1 c1(C(=O)NC2C(NC(C(C)N(C(C)=O)C)=O)C2)noc(-c2ccccc2)c1C C1(SC)CN(C(=O)CN(C2CCS(=O)(=O)C2)C)CC1NC(C1CC(C)CCO1)=O C#CCC(CC(=O)NCCc1cc(C)[nH]n1)NC(=O)C(C)C(C)C N1(C(C2CN(C)C2)=O)CCC2CN(C(c3cc4c(s3)CCSC4)=O)CC2CC1 Cc1ccc(CN(C(c2cc(C#N)ccn2)C(=O)NC2CCCC2)C)cc1Cl C(=O)(C(C)(C)CC1CCCCC1)NC(C(C)NC(CN(C1CC1)CC)=O)CO C1(NC(c2c(CC)occ2)=O)CCN(C(=O)CCSc2nccn2C)CC1C c1(C(CC)N(C(c2cccnc2)C(=O)NC2CC2)C(C)C)ccccc1 CC(C(=O)N(C)CC1CCCCN1C(C1(F)CCCC1)=O)C(F)F C1(N(C(C=CC(N)=O)=O)CC2CC2)CCN(C(c2snc(Cl)c2Cl)=O)CC1 c1(N2CCC(OCCNC(c3cc(C(C)C)n[nH]3)=O)C2)ncnc2cccc(F)c12 CC(C)CC(C(N)=O)N(C)C(C1CN(C(C2(C)CCCC2O)=O)CC12CC2)=O CC1CCCC1C(=O)NCC(C)(C1CC1)NC(c1nncn1C1CC1)=O CS(=O)(=O)c1ccccc1C(=O)NC1CCC(NC(c2cnns2)=O)CC1 n1(CC)cc(C(=O)NC2CC(CCNC(c3cc(C(C)(C)C)n[nH]3)=O)C2)c(C)n1 C(=O)(C1=CCCOCC1)NCCc1c(CNC(C2CC(C)OC2)=O)nco1 C(=O)(CC(C)CC(=O)NCCCNC(c1nc(Cl)c(Cl)s1)=O)OC c1(C(=O)NC(C2CCCCC2)CNC(C2(CSC)CCC2)=O)ccsc1Cl C1(C(=O)OCC)CCCC1ONC(C1CCC(C(F)(F)F)O1)=O C1(C(=O)NCCN(CCOC)C)CCN(C(=O)C=Cc2ccccc2)CCO1 C1(C)(C(N2CCCC(CC)C2)=O)CCN(OC(C=C2CCOC2C(=C)C)=O)CC1 N1(C(C(CC=C)CC=C)=O)CCCC2(CCC2NC(C2CC3C=CC2CC3)=O)C1 C(C(C)(O)CC(=O)N1CCC(C=CC(=O)NCCCCC(N)=O)CC1)OC CC1(C)CC(C(=O)NCC23CC2CN(C(=O)C2=C(Cl)CCC2)C3)C(C)(C)O1 N1(C(CC(CC)C2CC2)=O)CCOC(C)C1C(=O)NCC1(COC)CCC1 c1(CCC(=O)NC(C(=O)NCC(COCC)C)C2(O)CCC2)cnn(C)c1 c1(OC)ccc(C=CC(=O)N(CC(C)NC(=O)CCCC(C)C)C)cc1O C=CCC(C)C(=O)NC1(CCNC(=O)C(F)(F)C2(OC)CCC2)CC1 Cc1ccc2[nH]c(C(N3CCC4CC4(NC(=O)C(Cl)=CCl)CC3)=O)cc2c1C n1(CC#C)ccc2nc(Cl)nc(N(CC)Cc3cccnc3C(F)(F)F)c12 C(=O)(C(O)CCCNC(=O)OC(C)(C)C)N(C(C)(C)C(F)(F)F)C1CC1 C=C(C)CCC(=O)NCCCN(C(=O)C(CC=C)c1ccccc1)C1CC1 N1(C(C(CC(C)C)NC(c2nc(CC)oc2)=O)=O)CCC2CCC(C2)C1 C1(C(=O)NCC(C)(C)Cn2cc(CCN3CCCC3)nn2)CCCC1C1CC1 c1(C(N2CC3(CN(C(CCC)=O)C3)C2)=O)cnc2[nH]c(C(F)(F)F)nc2c1 c1(C(N2CCCCC(CNC(C3CC3(F)F)=O)C2)=O)cc2ccnn2cn1 N#Cc1ccc(NC(C2CC23CN(C(c2occc2Br)=O)C3)=O)c2ccccc12 CC1(C)CC(NC(=O)CS(C)(=O)=O)CN(C(c2cc3c(s2)CCC3)=O)C1 C(=O)(CCCC(=O)N1CCC(F)(CNC(C2CC3(CC3)CO2)=O)C1)OC(C)(C)C c1(C(=O)NC2CN(C(CCCC)=O)CC3C2C3)c(OC)cnc2ccccc12 c1(-c2cncc(C)c2)cnn2cc(C(=O)NC(c3ccc(Br)cn3)C)cnc12 C=C(C)CCC(=O)N1CC(CNC(=O)CC2CCOC(C(C)C)C2)C(C)C1 c1(NCC(C)OCC=C)ccc2c(S(N)(=O)=O)cccc2c1 C=CCC(CC=C)C(=O)N1CC(C2CC2)OC(C)C1 C1(C(N(CCCN(C(=O)CNC=O)C)C)=O)CC2(CC2)CO1 C12(C(N(CCN(C(=O)CC3C=CCC3)C(C)C)C)=O)CCC(C)(C1)OC2 C(c1cn(CCC#N)c2ccccc12)=CC(N1CCCCC1C1(NCCCl)CC1)=O c1(CC(CSC)NC(N2CC3CCCC23)=O)cc(F)cc(F)c1 C12(C(=O)NCC3N(C(C(c4ccc(C)cc4)=O)=O)CCCC3)CCCC1C2(F)F N1(C(c2c(C)snn2)=O)CC(CC(=O)NCc2csc(O)n2)CC1C C1(C(N2CC(NC(C(=O)NCC)=O)(CO)C2)=O)CCC2(CCC2)CO1 c1(C(N(C2CCN(C(=O)Cc3cscn3)C2)C)=O)ccc2nc(O)[nH]c2n1 CCCCCC(C)(C)C(=O)N1CCCC(CCNC(C2CCCCCCC2)=O)C1 c1(C(N(CC(=O)NC(CC)COC)C2CCC2)=O)ccc(C)cc1C N1(C(C2CCCC23CCC3)=O)CCCC2CCNCC12 N1(C(C(=Cc2ccco2)C)=O)CCC2CC2(NC(=O)C=Cc2csc(C)n2)CC1 C1(CCNS(NC(C)C)(=O)=O)CC12CCC(c1ccccc1)CC2.c1(=O)c(=O)[nH]1 CCCS(=O)(=O)CC(=O)NCCC1CCC(NC(=O)CSc2ccccc2F)C1 C1(C(=O)NCC(COC)O)CC=CCN1C(=O)CC1(OC)CCC1 N1(CC(=O)NC(C)C(N2CCCCC2)=O)CCc2ccccc2C(C)C1 C1(NC(C2CCCS2)=O)CC12CCN(C(=O)CCC1CC1(F)F)C2 C1(NC(C(CSC)(C)NC(c2ccsc2C)=O)=O)CCCOC12CCC2 C(=O)(CC(C(F)F)NC(c1cc(O)ccc1F)=O)NCC(C(C)(C)C)O C1(NC(CSCCC)=O)CCCCN(C(C2CCC2C(C)(C)C)=O)C1 c1(-c2nc(C(CCC)C)nn2Cc2cccc(OC)c2)cc(F)cc(F)c1 c1(CNC(c2cc(O)ccc2F)=O)nc(CNC(C2CCCCS2)=O)cc(O)n1 C1(CNC(C=C2CCC(C)C2)=O)CN(C(=O)Cc2cnn(C)c2)CC2(CCC2)O1 C1(F)(CNC(=O)CCc2cccnc2)CCC(NC(=O)CCc2cnc[nH]2)C1 CC1(F)COCCN(C(C2COCCN(C(c3cccc4nccn34)=O)C2)=O)C1 N1(C(C(C)c2cc[nH]n2)=O)CC(C(=O)NC2(C)CCCOC2)C2(CCC2)C1 CCCC(C(=O)NC(CNC(=O)Cc1csc2ccccc12)CCOC)C(C)C CN1CCC(O)C(NC(C23CC(CN(C(=O)CNC(=O)C4CC4)C2)C3)=O)C1 C1(C)(CS(N2C(C(=O)OC)CC2CO)(=O)=O)CCCCC1(F)F CN1CCC2OCCN(Cc3nc(-c4cnn(C)c4)nn3C3CC3)C2C1 C(=O)(C1=CCCC(C)(C)C1)NC1CN(C(c2n(C)nc([N+](=O)[O-])c2)=O)C1 S(=O)(=O)(c1ccc(F)c(Br)c1)N1C(C)(C(=O)Nc2cc(I)cnc2Cl)CC1 C1(N(C(C(C)NS(C)(=O)=O)=O)C)CCN(C(c2sccc2C(=O)OC(C)(C)C)=O)C1 N1(c2cc(C)nc(C(F)(F)F)n2)CCn2ncc(CNC(=O)C(C)O)c2C1 C1(NC(=O)C2=C(Cl)CCC2)CCCC12CN(C(=O)C=Cc1cnc(O)nc1O)C2 c1(CC)nc(C)c(C(=O)NC2C=CC(CNC(=O)CCP(C)(C)=O)C2)c(C)n1 C=C(C)c1ccccc1NC(=O)C(C1CCCN(C(C2CC=CCC2C)=O)C1)C C1(C(N2CCC(OCC(N)=O)C2)C(=O)NCCC#N)CC2CCC1CC2 N1(C(C2(CC=C)COC2)=O)CC(NC(C2CCCOC2)=O)CC2(CC2)C1 CN1CCC(C(=O)NC2C=CC(CNC(=O)CCCn3ccccc3=O)C2)CC1 c1(OC)cc(C(=O)NC2C(N(C)C)CN(C(C3(OC)CC3)=O)C2)ccn1 c1(N2CCCC(OC)C2)nc2ccc(Cl)cc2c(=NCC2CN(C)CCO2)[nH]1 C1(C(N(C(CC)CC)CCO)=O)CC2(CC(NC(C3CC4CCC3CC4)=O)C2)C1 N1(C(C(C)C2(O)CCC2)=O)CCCC(O)(CNC(=O)Cc2cn[nH]c2)C1 C1(NC(C(CC)NC(C)=O)=O)CCN(C(=O)C(C)CNCC)C12CCC2 Cc1n[nH]c(C)c1C(C)C(=O)NCCC1(CNC(C2CC3C=CC2C3)=O)CC1 CCC(CC)(CCNC(c1ncccc1N)=O)NC(=O)CC1CCCCC1(F)F C(CN=c1[nH]c2c(c(=NC(C)CCC(C)C)[nH]1)COCC2)c1scc(CC)n1 CCCCCC(C)(C)C(=O)N1CCCC1CN1CCC(=O)NC(C2CC2)C1=O c1(CC(=O)NC(CNC(C2C(C)(COC)C2)=O)C2CCC2)cc(C(F)(F)F)n[nH]1 C1(C(=O)OC)CCN(C(c2cncc(OC(C)C)c2)=O)C12CCSCC2 CCCC(C(=O)N1CCC(NC(=O)CNS(C)(=O)=O)C1)NC(N)=O C1(C(=O)NC(CC(C)NC(c2c(CC)nc[nH]2)=O)C)CCc2ncncc2C1 C1(NC(CC(CC)(F)F)=O)CC2CC(C1)N(C(=O)CC1CCSCC1)C2 C1(NC(=O)COCC2CCOC2)CCN(C(c2cc(CO)on2)=O)CC1F c1(OC)cccc(CC(C(=O)Nc2nc(C)cs2)NC(=O)OC(C)(C)C)c1 CS(=O)(=O)C1CC(C(N2CCC(NC(=O)CCc3cc(Cl)no3)C(F)C2)=O)C1 CCCCC(CNC(c1ocnc1CC)=O)NC(c1ccc(-c2ccco2)o1)=O N(C1CCc2cccnc21)C(C1CC(C)(C)N(C(=O)C(=O)C2CCCC2)CC1)=O C(=O)(C(C(C)(C)C)N1CCCCC1=O)N1C2C(NC(C(CC#C)C)=O)C(C2)C1 c1(NC(CC(CNC(C(CCC)CC)=O)C2CCC2)=O)ccc2ncnn2c1 C(C(C(=O)NCC(F)(F)F)NC(C1CC(C)(C)C1)=O)OC(C)C S(=O)(=O)(c1ccc(Cl)c(NC(NC2CCn3ccnc32)=O)c1)NCC=C c1(NC(=O)NC)cc(Br)sc1C(=O)N(C1CCN(CC)C1)CC(N)=O c1(C(N2CCC3(NC(c4cc(SC)oc4C)=O)C(C2)C3)=O)nc(C)c(C)[nH]c1=O C1(CC(=O)NC2CC(C(C)O)C2)CCCN1C(=O)CC1CC(F)(F)C1 N1(C(C(C(CC)C)C)=O)CC2(C1)C(NC(c1ccco1)=O)CCS2(=O)=O C=CC1(CC(=O)NCCC(O)CCC)CN(C(c2cnn(C)c2Cl)=O)C1 N1(C(=O)CC2CCC2)CC2OCCN(C(C3CCN(NC(CC)=O)C3=O)=O)C2C1 C(c1ccc(Cl)c(Cl)c1)=CC(=O)NC1CC(C(=O)Nc2ccc(I)cc2Cl)C1 Cc1cccc(C(=O)NCC2CN(C(=O)CC3CCCCCO3)CCO2)c1 C1(CC(N2CC(C(=O)NC)C2)=O)N(C(C2(C(N)=O)CCC2)=O)CCC1(C)C c1(C(N(CCC)CCNC(C2(C3CC3)CCC2)=O)=O)cnc(Br)c(O)c1 c1(C(=O)NC2(CF)CCN(C(C(F)=CC)=O)C2)cc(=O)c2ccccc2n1C c1(CCNC(C(=O)NC2C(CC)COC2)=O)cn(C(C)(C)C)nc1C N1(C(C(CCC)OC)=O)C(C)CC2CN(C(c3cccc4oc(=N)[nH]c34)=O)CC12 CC(CCN(C)C)C(=O)N(c1ccccc1)C(c1cccnn1)=O C1(C(N2CCC(COC)(NC(=O)CC3CCC4CC4C3)C2)=O)CNC(=O)CC1C C12(NC(COCCOC)=O)CCCCC1N(C(=O)CCOC1CCC1)CC2 n1(CC(=O)OCC2CC(OC3CCC3)C2)cc(C(F)(F)F)cc(Br)c1=O n1(CCC)nc(C)cc1C(=O)NCC1(O)CN(C(=O)C(C)Cc2ccco2)C1 N1(C(c2c(CC)scc2)=O)CC(NC(C2(CF)CC(F)(F)C2)=O)C(C2CC2)C1 Cc1ccc(C(=O)N(CC(C)(C)NC(=O)Cc2ccnn2C)C)c(Cl)c1C c1(N2C3CCC(NC(Cc4cc(C)[nH]n4)=O)C(C3)C2)ncnc2ccc(Cl)cc12 C(=O)(CC(F)(F)Cl)N(CCN(C(C(c1ccc(CC)s1)=O)=O)C)C(C)C c1(CNc2cccc(C(=O)Nc3cc(SC)n[nH]3)c2)cc(O)cc(O)c1 C1(C(N2CCC(NC(C3CN(CC(C)C)C3)=O)C2)=O)C(F)(F)C12CCC2 N1(C(c2c(C(C)C)scn2)=O)CCCC(CCNC(=O)C(C)(C)c2ccns2)C1 c1(C(=O)NCC2CCC(CNC(c3cc(C)oc3C)=O)CC2)cc(Cl)nc(Cl)c1 N1(C(C(CC)CC(C)C)=O)CCCC2(CCCN2C(c2cc3scnc3[nH]2)=O)C1 C1(NC(c2c(COC)ncs2)=O)CCN(C(=O)CS(=O)(=O)NC2CC2)CCC1CO N1(C(C(n2c(C)cc(C)n2)C)=O)CCC(C)(CNC(C23COCC2C3)=O)CC1 N1(C(=O)OC(C)(C)C)CCC(C2CCC2)(C(=O)N=c2cc(CCOC)[nH][nH]2)C1 C1(C(=O)NCCC(C)NC(=O)C(F)(F)Sc2cnn(C)c2)CC2(C1)CC2F N1(C(c2ccc(CCC)[nH]2)=O)CCC2CC(C1)CN(C(=O)CC(C)CN(C)C)C2 N1(C(C2C(C=C)CC2)=O)CCCOC(CNC(c2nocc2CC)=O)C1 c1(CC)ccc(Br)cc1C(=O)NCC(CNC(c1cc(C)ns1)=O)OC CCCC(C(=O)N(CC(C)NC(=O)CC(c1ccccc1OC)C)C)N(C)C CC1OC(=O)NC1C(N1CCCC1CC(=O)Nc1ccccc1CCO)=O N1(C(CS(CC)(=O)=O)=O)CCOC2CCN(C(C3CCC4CC34)=O)CC12 C=C1CC(C(=O)NCC2CCC2)(COC)C1.C1CN(C(=O)CSCC2CCCO2)C1 N1(C(C(CCSC)OC)=O)CC2(NC(=O)C(=Cc3ccco3)C)CCCC2(F)C1 c1(CNC2CC(CC(N3CC(C#N)OCC3)=O)C2)c(Br)cc(Br)c(O)c1Br N1(C(c2cccc(C)n2)=O)CCN(C(C2CCC(=O)O2)=O)C(C(C)C)C1 N1(C(=O)CC2CCCO2)CCCC2(CCN(C(C34CC5CC3C4C5)=O)C2)C1 S(=O)(=O)(CC(F)(F)F)N1C(CC(=O)Nc2cnc(Br)c(F)c2)CCCC1 C1(C2CC2)(CNC(C2N(C=O)CCC2)=O)CCN(C(=O)CC=C(Cl)Cl)C1 C1(NC(C(CC#C)C2CC2)=O)CN(C(c2ccnc(CO)c2)=O)CCC12CCC2 CC(CF)CC(=O)NC1CC(NC(C2(OCc3ccccc3)CC2)=O)C1 c1(OC)cc(C(=O)NCC(C2CC2)N(C)C(c2ccco2)=O)c(C)cc1O C(c1cccc(F)c1Cl)=CC(=O)NC(CNC(c1c(C)oc(Cl)n1)=O)(C)C c1(CC)cc(C(=O)NCCc2ocnc2CNC(=O)Cc2nc(C)cs2)ncn1 C(=O)(CCC(O)C(C)(C)C)N1CC(C(=O)OC)C(c2ccccc2)CC1 CCC(F)(F)CC(=O)NCC1CN(C(c2cccc(CO)c2)=O)CC1(C)C c1(C(=O)NCC2CCCN(C(C(CNC(C)=O)(C)C)=O)C2)c(Cl)cncc1Cl c1(OCC(=O)NCC2(NC(=O)CCc3cnn[nH]3)CCOC2)cc(F)cc(Cl)c1 Cc1cc(C)c(C(=O)NCC2CCCN2C(C23CCN(CC2)CC3)=O)c(C)n1 C=CCC(CNC(=O)CC1CCC=CCC1)C(=O)NC1CC(C)(CO)C1 N1(C(C2CCCC(O)C2)=O)CC2COCC2(C(N2CC3OCC(CO)C3C2)=O)C1 c1(NC(CCC)C(=O)OC(c2ccccn2)C)cc(Cl)c(NC(=O)O)c(Cl)c1 CC1=C(C(=O)NC2(C)CC(NC(C3CC3c3c(F)cccc3F)=O)C2)CCO1 c1(C(N2CC(NC(C(C)c3cccs3)=O)C(O)C2)=O)cc2cccnc2cn1 N1(C(C(C(CC)O)C)=O)CC(C2CCCN(C(=O)CCc3ccsc3)C2)C1 N1(C(C2CN(C)C2)=O)CC(CNC(C2(CC3CC3)CCCO2)=O)C2(CCC2)C1 CCCCCCC(C)(CC)C(=O)NCC1CC2COCC2N1C(=O)CCCC#N C(=O)(CC(C)C(C)(C)NC(c1nc(C)ccc1F)=O)NCC(C#C)C(C)C c1(C(=O)NCCCN(C(C=NOC)=O)C2CC2)cnc(O)n(C2CC2)c1=O C(CN=C(NC1CC1)N1CCCC(n2ccnn2)C1)c1cccc(Cl)c1 C1(C(=O)NC(CC(=O)OC)C)CCCCCN1C(=O)C(=O)N(C)C n1(CC(=O)NCC2CN(C(CS(=O)(=O)NC)=O)C2)c(C)cc(C)nc1=O C(=O)(C1CCc2ccccc21)NC1CCCCN(C(c2c(C)nncc2)=O)CC1 N1(C(CCSCC(C)C)=O)CC(NC(C2(C)CC2c2ccccc2)=O)C(C)C1 C1(CN(C(C(=O)NCC)=O)C)CCCN(C(C2CC(SC)C2)=O)C1 CC1(C(=O)NC2CCC(CNC(=O)CCC=CC(=O)O)CC2)COCCO1 C(C(C(=O)NCC1CCOCC1)NC(=O)OC(C)(C)C)SCC c1(C(N2CCN(C(C(C=C)O)=O)C(C)C2)=O)c(OC)cc(OC)c(Cl)c1N c1(C(=O)NCC2CN(C(C3CC(CF)C3)=O)CCO2)cccc(C#CC2CC2)c1 CC1(C)CN(C(c2ocnc2C(F)F)=O)CC1NC(=O)CC1CCC(=O)NC1=O N1(C(C(Cc2ccccc2Br)NC(CC(C(C)C)O)=O)=O)CC(O)(C2CCC2)C1 N1(C(c2ncc(C)nc2)=O)CCC(NC(c2nccnc2Cl)=O)C(F)C1 C(CNC(c1ccccn1)=O)(C(C)(C)C)NC(C(C)(C)NC(=O)NCC=C)=O C1(CNC(CCc2cn(C)nc2)=O)CC(F)CN1C(=O)CO N1(C(C2C(C)(CC)C2)=O)CCCC(CO)(NC(=O)CC2(O)CCCN(C)C2)C1 c1(C(N2C(C)(C(=O)Nc3ncn(C)c3)CC2)=O)ccc(S(C)(=O)=O)cn1 c1(C(=O)NC(CC)CNC(=O)Cc2cocn2)ccc2n[nH]cc2c1 C1(CNC(CCNC(C)=O)=O)CC2(CCN(C(c3cc(F)cc(Br)c3)=O)CC2)C1 c1(OC(C(=O)N(CC(C)NC(C(CCC)C)=O)C)C)ccc(C#N)cc1 C1(C(N(C(C2CCC2)C)C2CC2)=O)Cc2ccccc2CN1Cc1ccccc1 N1(C(C(CNC(c2ncc(Cl)cn2)=O)N(C)C)=O)CCOCC(CO)C1 CC1=NN(C)C(=O)C1CC(=O)NCC1(CNC(c2cccc(O)c2Cl)=O)CCC1 C(C(C)(C)CC(C)O)NC(C1(NC(CCN(CCC)C)=O)CSC1)=O c1(C(=O)OC)nc(N2CC3CC3(CNCC3(c4ccccc4)CC3)C2)ncc1F N(C1CCc2cccnc21)C(C(c1cccnc1)NC(c1n(CC)ncc1)=O)=O N1(C(C2=C(C)CCC2)=O)CCC2C(CCN2C(c2coc3ccc(F)cc23)=O)C1 CC1CCCC1(C(=O)NC1CC(CCF)C1)NC(c1cc(C2CC2)on1)=O c1(OC)ccnc(CC(=O)NC2(CCCNC(c3n[nH]cc3OC)=O)CC2)n1 C1(NC(=O)CCc2cnn[nH]2)CC(O)CN(C(=O)CN2CSCC2=O)C1 c1(C(=O)NC2(C)CCN(C(C3(C4CCCCO4)CC3)=O)C2)ccc(Cl)c(O)c1N C1(C(N2CC(CCNC(C(C)(C3CC3)OC)=O)C2)=O)CNC(=O)CC12CCC2 N1(C(C(CC)N(CC)CC)=O)CCC(C2CC2)(CNC(C2(OC)CC2)=O)C1 C12(CNC(=O)NC3(Cc4ccccc4)CCOCC3)OCCCC1C2(F)F N1(C(c2cc(-c3ccccc3Cl)no2)=O)CC2C(CNC(C3(CF)CC3)=O)C2C1 c1(NC(COC)C(C)C)nc(N2CC(=O)N3CCCC3C2)c2sccc2n1 CC(CC(=O)NCCOCCC(=O)NCCc1nccs1)n1cccc1 C1(O)(CCNC(=O)CSc2ccncc2)CCN(C(=O)Cc2cncnc2)CC1 N1(C(COCC=C)=O)CCC(C)C(N(C)C(c2cc(C(=O)OC)no2)=O)C1 c1(N(CCN=c2cncc[nH]2)C)cc(Br)ccc1S(=O)(=O)NC1C2CCCOC12 c1(C(N2CCC(C(C)NC(c3ccon3)=O)C2)=O)cc(F)c(N)cc1F c1(CC)cc2c(CC(=O)NC3CCC(NC(=O)C(C)C(F)F)C3)csc2s1 N1(S(C)(=O)=O)CCCCC1C(=O)NC1C=CCN(C(C2(O)CCC2)=O)C1 N1(C(C(C(C)C)NC(C)=O)=O)CCCC(NC(=O)COCC2CCCC2)C1C C1(c2cn(C)nc2)CC1N=c1[nH]c(=NC2CCSCC2)[nH]c2ncn(C)c12 C1(C(=O)NCc2c(CCNC(C(C3CCC3)OC)=O)ocn2)CCC(C)(C)CC1 c1(OC)ccc([N+](=O)[O-])c(NC(=O)CC2CN(C(c3ccsc3OC)=O)C2)n1 C1(NC(CCCCCC#C)=O)CCN(C(=O)CC2CCC3CC3C2)CC12CCC2 O=C(CCCNC(=O)CC1CCN1C(=O)CC1CC2C=CC1C2)NO C1(C(=O)NCC2CCC(NC(=O)COC3CCOC3)C2)CC12CCS(=O)(=O)CC2 C(C(C)C(F)C(=O)NCCN1CCC2CC12)NC(Cc1c(C)ccnc1)=O C(CCCCC(=O)N1CCC(C(C)(C)NC(c2csc(C#N)c2)=O)C1)=CC C1(CC(=O)NCC2C(CNC(=O)Cc3cnns3)C2)CCCCO1 C(=O)(C1=CCCCC1C)NC(C(C)C)CCN(C)C(c1nc(C2CC2)cs1)=O CC1=C(C(=O)NCC2(C(C)(C)O)CN(C(=O)CC3CCCN(C)C3)C2)COCC1 n1(C(c2c(C)cccc2)c2nc(-c3cscn3)nn2C)c(=O)oc2ccccc12 c1(C(=O)OC)cc2[nH]c(C(N3CC4CC(NC(=O)CCS(C)=O)C4C3)=O)cc2s1 C12(C(=O)NC3(C)CCCN(C(C4(C)CCCCO4)=O)C3)CC3CC(C(=O)N1)C2C3 C(=O)(C1=NOC(C)C1)NC1(c2ccccc2)CN(C(c2n(C(C)C)ccn2)=O)C1 C1(F)(CNC(CCSC)=O)CCC(CNC(=O)CC2CCCC(O)C2)CC1 Cc1cc([N+](=O)[O-])cc(C(=O)NCCC(O)CNC(=O)Cc2ccoc2C)c1Cl N1(CC(=O)NC(c2cn(CCCC(=O)NCC(F)(F)F)nn2)C)CCOCC1C C(=O)(C(O)C(F)F)N(CCNC(c1ccc(O)nc1)=O)C1CC1 c1(NC(c2cc(C)c(Oc3ccc(F)cc3)cc2)=O)ncc2c(n1)COC2 C(CO)(CCCCNC(=O)C(O)C1CC1)NC(c1c[nH]nc1[N+](=O)[O-])=O CS(=O)(=O)c1cc(NC(=O)Cn2cc(COC3CCOC3)nn2)co1 N1(C(c2occ(C(C)=O)c2)=O)CCC(CO)(NC(=O)CC(C)c2ccco2)C1 c1(C(=O)Nc2c(C#N)ncn2-c2ccccc2)cc(-c2cnoc2)cc2[nH]ncc12 c1(C(N2C3CN(Cc4ccc(C#N)cc4)CC2C3)=O)cc2cn[nH]c2cn1 c1(CC)nn(C)cc1C(=O)NCCCC1CCCCN1C(C1CC(=O)N(C)C1)=O C12(NC(C=C(CC)CC)=O)CCN(C(c3ccc(OC(F)(F)F)nc3)=O)CC1C2 c1ccc2c(c1)OCC2CNc1nccc(N2CCC3(CCSC3)C2)n1 N1(C(C(CC)NC(c2ccc(Cl)cn2)=O)=O)CCC(C)(C(C)C)CC1 c1(C(C)C)cc(C(=O)NCC(CO)NC(=O)Cn2ccnn2)ccc1F c1(C(=O)NC2(C)CCN(C(C3(C)CCC3)=O)C2)ccc(Br)c(O)n1 C1(C#N)(C(N2CCC(C)(C(=O)NOCCCN(C)C)C2)=O)CCCCC1 C12(NC(c3ccnn3C3CC3)=O)CCN(C(=O)CSCc3ncc[nH]3)CC1C2 Cc1ccc2c(c1)SC(C(N1CCC(NC(c3cccnc3)=O)C1(C)C)=O)C2 C(=O)(CCC(=O)N1CCC(O)CC1)NCCC(C)N(C)C(C1CCO1)=O c12cnn3c1CC(CC3)N2.C1(CC(=O)NC)CCN1C(=O)OC(C)(C)C c1(C(N(C2(C(N(C(C)CC(N)=O)C)=O)CC2)C)=O)ccc(=N)[nH]n1 N1(C(c2cn(C)cc(Br)c2=O)=O)CCN(C(=O)CNC=O)CC(C)(C)C1 C(N=c1cc(C)[nH]c(=NCc2nccn2-c2ccccc2)[nH]1)C1CCC(=C)CC1 CC1CC(NC(=O)CCSC(F)(F)F)CCN1C(C1CCCSC1)=O C(CCC(=O)N1CC(CCO)C1)(C(C)C)NC(C1C(CC)N(C)CC1)=O C1(N(C)C)CCN(CCC(N2CCCC2c2ccc(C(=O)O)nn2)=O)CC1 N1(C(CC(CC)C)=O)CC(NC(=O)C2=CCCSC2)C2CC2C1 c1(OC)ccc(C(N2CCC(CN(C)C(C3CC3C)=O)C2)=O)cc1S(C)(=O)=O c1(C(C(=O)NCCNC(C(C)OCCCCCC)=O)O)cccc(Cl)c1 C1(NC(Cc2ccc(OCC)cn2)=O)CN(C(c2csnn2)=O)CC2CC12 C(=O)(CC(C)C(F)(F)F)N(C(C)C(=O)NC(CO)CCO)CC c1(CC(=O)NCC2CCN(C(CCC(CC)C)=O)CC2)ccc2c(c1)CCC2 C1(C(N2CC(C)C2(C)C)=O)CC(N=[N+]=[N-])CN1C(C1CCNC1=O)=O c1(C(C)=O)ccc(C(N2CCC(O)(CNC(=O)C=Cc3cnccn3)C2)=O)nn1 C1(C(=O)NCC2(O)CC(NC(c3cncc(N)c3)=O)C2)CCc2nccn2CC1 N1(C(c2cc(CNC(c3cn(CC)nc3C)=O)[nH]n2)=O)CC2CC(C)C2C1 C#CCCCC(C)C(=O)NCC1CN(C(C2CCCN2C)=O)C1 C(=O)(CC(C)C(F)(F)F)NC(CCSC)C(=O)NCc1cc(F)ccc1O C1(CC)CN(C(c2cccc(C(C)C)c2)=O)CCN1C(=O)C=C1CCN(C)CC1 CC(CO)CCN=c1[nH]c(N2CCC3(CC2)CN(C)C3)nc2c1CCC2 C1(C(=O)NC(CCNC(C2CC(=C)C2)=O)C)CCC(C)(C)O1 c1(-c2n(-c3ccc(C)cc3C)nc(-c3ccccn3)n2)cc2cc(Br)ccc2s1 C(=O)(CCCCCO)N1CCC(C)C1CNC(=O)C(c1cncn1C)O c1(OC)nscc1NC(c1nnnn1CC1CC1)c1nc[nH]n1 c1(C(N2CCN(C(c3cc(C)ncc3C)=O)C3C2C3)=O)cc2ccccn2c1 Cc1sc(C(N2CC(CO)(NC(=O)C=CC3CCOC3)C2)=O)c(C)c1C C1(NC(=O)Nc2ncnc(OC)c2OC)CC2CCCCN2C1 CCC(C)(C)C(=O)C(=O)N1CCC(CNC(=O)CC2CCC(O)C2)C1(C)C CN1CCN(C(=O)CCc2cn[nH]c2)CC1C(=O)Nc1cccnc1 CCC(C)(C)C(O)C(=O)NCCN(C(=O)C=CC(C)CC)C1CC1 c1(CC(=O)NC2CCN(C(C(C(C)C)SCC)=O)C23CC3)cccc([N+](=O)[O-])c1 C1(OCC(=O)N(CCCNC(C(C)=CC)=O)CC)CCCCC1C CC(Cl)(Cl)C(=O)N1CCC(CCNC(=O)C(O)COCc2ccccc2)C1 c1(C(N2CCN(C(=O)NC3CCNCC3)CC2)=O)ccccc1Cl N1(C(C(C(C)OC)NC(=O)C(C)S(N)(=O)=O)=O)CCC2(CC1)CC(O)C2 CCC(C)CC(=O)C(=O)NCCn1ccc(C(=O)NCCN(C)C2CC2)c1 c1(C(=O)NCC2(NC(=O)CC3CSCCS3)CC2)cncc2c1CCCC2 CCC(CC(=O)NC1CC(OC)C1)N(C)C(c1cccc(O)n1)=O c1(C(=O)NCCC(CNC(c2cscc2Cl)=O)O)noc2cc(F)ccc12 C#CC1(O)CCN(C(=O)CC2CCC(NC(=O)CC(C)CC(=O)OC)C2)CC1 C1(O)(c2cn(Cc3cccc(C)c3)nn2)CCN(C(C2CCC(=O)N2)=O)CC1 C1(CNC(=O)C(O)Cn2cncn2)CC(O)CN1C(c1ccc(Cl)o1)=O C(CN=c1nc(C)cc(C)[nH]1)C1N(C(C(c2ccc(C)cc2)C)=O)CCCC1C c1(C(N(CCCN(C)C(C2(C)CCCO2)=O)C)=O)ccc(N)cc1O C1(N=[N+]=[N-])(C(=O)NCC(C(CC)C)CO)CCN(C(=O)CN2CCCC2=O)C1 Cc1ncncc1C(=O)NCC1CCCN1Cc1cccc(-n2ccnc2)c1 CON=CC(=O)NC1(CCNC(=O)CC(=O)NC(C)C)CC1 c1(NC(C)=O)cc(C(N2CCC2CNC(=O)C(C)CF)=O)ccc1[N+](=O)[O-] N1(C(C(CC=C)CNC(c2cccc(OC)c2)=O)=O)CCC(C)(C2CC2)C1 C(CCCS(C)=O)OC(=O)C(F)CC1CN(C(=O)OCC)C1 CCCCC(CC(=O)NCc1noc(C(N)=O)n1)NC(C1(C)SCCCS1)=O C1(NCC(N2CC(CCO)(NC(C(C)OCC)=O)C2)=O)CCCCC1N(C)C c1(C(N2CCN(C3CCN(C(C)C)C3=O)CC2C)=O)cnn2ccccc12 c1(C(=O)NCC(=O)NCC(CNC(C2CCCCS2)=O)OC)cc(F)cc(F)c1 C1(F)(CNC(CNC(C)=O)=O)CCCN(C(c2cc(OC)c(C3CC3)nn2)=O)C1 C1(C(N2CCC(CCNC(=O)C=Cc3cnccn3)C2)=O)CC2COCC2C1 n1(CC(=O)NCC(C2CC2)NC(C(N2CCSCC2)C)=O)cnccc1=O N1(C(CCC(=O)NC)=O)CC(C)C(NC(c2cnn(C)n2)=O)C(C)C1 S(=O)(=O)(c1ccc(C(=O)N(C(CC)C)C)cc1)N1Cc2ccc(cc2)C1.NC C1(C(C)(C)C)(CNC(C2CCCCC2c2nc[nH]n2)=O)CCN(C(=O)CCl)C1 C1(CNC(C2(NC(=O)CC3CC3)CSC2)=O)CC(CO)CO1 C1(CNC(C(n2cc(-c3ccnn3CC(F)F)nn2)C)=O)CCCCC1(F)F C1(C(=O)NC2C(NC(CCSCCC)=O)CCOC2)CCCCCS1(=O)=O C(=O)(C1=CC(C)CC1)NC1CCC(NC(Cn2c(C)c(Cl)cn2)=O)C1 C(=O)(CCCCC(N)=O)NCC(CC(=O)NCCC(O)C1CCC1)OC CN1CCC(NC(=O)C(CC(F)F)NC(C2CCN(C)C2)=O)C1(C)C C1(CCOC)(OC)CCN(C(=O)CCCN2CCCC2)C1.C(C1C(=O)N1)OCC CC1(C(N2CCC(C)(NC(=O)COc3cccnc3)C2)=O)CC(C(F)(F)F)=NO1 CN1N=C(CC(=O)NC2COCC2NC(c2ncnc3c2CCCC3)=O)CC1=O CC1COCC(C(N2CC(F)CC2CC(=O)NC2CC2C(F)(F)F)=O)O1 N1(C(c2c(OC)nsc2OC)=O)CC(C)CN(C(c2ccc(C)c(F)c2)=O)C(C)C1 C1(NC(CCC2N(C(CC(C)O)=O)CCC2)=O)CC(F)(F)C1(C)C c1(SC)cccc(CC(=O)NCC2(C)CCN(C(c3cn(C(F)F)cn3)=O)C2)c1 C1(C)(CC)CCC(C(=O)NCC#CCNC(=O)C(F)(F)C2CC2)O1 c1(C(N2CCC(N(C(c3nn(C)cc3Cl)=O)CC)CC2)=O)c(O)nnc(C)c1C C1(C(=O)NC(CCC=C)C)CN(C(=O)CC(C)C(F)(F)F)CC12CCC2 Cc1nnc2ccc(C(=O)OCCc3nnc(C)n3C)nn12 Cc1ccc(C(N2CCC(F)(C(=O)Nc3cccc(F)c3C)C2)=O)c(C)c1 CN1CCCC(C(=O)NC2CC2NC(c2ccc(Cn3ccnc3)cc2)=O)C1 N1(C(c2ncn(CC)n2)=O)CCC2(CC1)CC2CNC(=O)C1=C(C)CC1 C1(CCC(=O)NCCCN(C(C2(CCF)CCC2)=O)CC)CCCN(C)C1 C1(N2CCN(C(c3nc(C(C)C)sc3)=O)CC2)CCCCNC1=O c1(C(N(CCCN(C(CC2CCN(C)C2)=O)C)C)=O)ccc(F)c(O)c1 N1(C(C(OC)OC)=O)CC2(CCC(CNC(=O)C(C)n3cccn3)O2)C1 c1(C(N2C(C(=O)NC3(C(C)C)CC3)CC=CC2)=O)c[nH]c2ncccc12 CC1(C)CN(c2cc(Cc3cnc4[nH]ccc4c3)ncn2)CCC1NC1CC1 c1(OC)cc(Cl)ccc1CC.C1(c2nc(C(N)=O)no2)CNCCO1 c1(CNCC2C(NC(C(C)SC)=O)CCC2)cc(O)nc(C2CC2)n1 S(=O)(=O)(c1ccc2c(c1)nnn2C)N1CCN(C)C(C2CCC2)C1 C1(C(NOCCCOC)=O)CCC(CNC(=O)C=C(C)C2CC2)O1 Cc1ccc(C(N2CCCCC2C(=O)NCC(C)(F)C(C)(C)F)=O)nc1O CN1CC=C(C(=O)NCCC2CN(C(C3CC(=O)N(C)C3)=O)CCCO2)C1 c1(CC)cncc(C(=O)NCC2CCCC2NC(c2ccc[n+]([O-])c2)=O)c1 c1(C(=O)NC2C3(CN(C(C(C)(Cl)Cl)=O)C3)CC2)ccc(F)c2ccccc12 C(=O)(N1CCC(C(=O)O)O1)C1CC(C(=O)NCC2CCCOCC2)C1 C1(C(C)C)CNC(=O)CN1C(=O)C(CNC(c1ccc(O)cn1)=O)CC1CC1 c1(C(N(CC(C)(C)NC(C2CN(C(N(C)C)=O)C2)=O)C)=O)cnc2c(c1)CCC2 c1(C(=O)NC(CNC(C(CCSC)OC)=O)C2CC2)coc2c1NC(=O)CCC2 n1(CC(=O)NC2(CF)CCN(C(C3CCC3(F)F)=O)C2)cc(Br)ccc1=O c1(N2CC3CC(NC(c4cncc(F)n4)=O)CC3C2)ccc(Cl)cc1[N+](=O)[O-] c1(NC(C(C)(C)F)=O)ncnc2c1CCO2.C(C1CC1)=CC N1(C(C(CCC2CC2)NC(c2cnc3cc[nH]c3c2)=O)=O)CCC(C2CCC2)C1 N1(C(=O)OC(C)(C)C)CC2(CCCCC2)C1NC(=O)OCCc1ccsc1Br c1(NCC2(OCC)CCC2)ccc(S(=O)(=O)N2CCN(C(C)CO)CC2)cc1Br N1(C(=O)Nc2ncc(C(F)(F)F)s2)CCC(c2cccs2)CC1 c1(NC=O)ccc(C(=O)NCC2CCN2C(c2ccc(-c3cnc[nH]3)cc2)=O)cc1 N1(C(c2cccn(C3CCC3)c2=O)=O)CCN(C(C2CC=CCO2)=O)C(C2CC2)C1 c1(CC)ccc(C(=O)N(C)CC2CC(F)CN2C(c2csc(COC)c2)=O)cc1 c1(C(=O)NCC2C=CC(NC(Cc3c(C)ncs3)=O)C2)cn(C)c(=O)cn1 Cc1cc(C#N)nc(N2CCCC(O)(CNC(C3(O)CC3)=O)C2)n1 C=CCCCCCC(=O)NCC1CC2CN(C(c3ccc4cc[nH]c4c3)=O)CC12 C1(CCC)(NC(=O)C(C)C(F)(F)F)CCN(C(c2ccc(C)cc2)=O)CC1 CC(C)(C)CCCC(=O)NC1CCCCC1n1cc(-c2c[nH]nc2C(=O)O)nn1 c1(N(C(=O)CSCC(N2COCC2(C)C)=O)C)ccc(F)cc1 c1(CNCC(=O)O)cccc(-c2cn(CCCCC(=O)NCC(F)(F)F)nn2)c1 c1(CNC(CCN(C)C(C2CCC2C(C)(C)C)=O)=O)nc(CC2CC2)cs1 C(CCC(O)CO)N(C)C(C1CC(CNC(=O)Cn2nccn2)C1)=O Cc1cncc(C(N2CCCCC2C2CCN(C(=O)CC3CCCCO3)C2)=O)c1 C(C)(CCCC(=O)N1CCOC(C(C)C)C1)NC(C1C(=C)C1)=O C1(NC(c2[nH]cc(C)c2)=O)CN(C(c2ccc(C#N)cn2)=O)CCC1O c1(C(=O)NC(COC)CC(=O)NCCc2ncoc2C)ccc(C)cc1C C12(NC(C3(C(=O)OC)CC3)=O)CC1CN(C(c1occc1Cl)=O)C2 n1(CC=C)c(N2CCN(c3ccc(OC)cc3)CC2)nnc1-c1ccc(O)nc1 C(C(CC(=O)NC1(C)CS(=O)(=O)C1)C1CCC1)NC(C1C(C)=CCS1)=O c1(C(c2nnnn2CCCF)NCC(COC)C)cccc(OC)c1C CC1CCc2nc(Cl)nc(N3C4CCC3CN(C(C35CC(CO3)C5)=O)CC4)c2C1 Cc1nn(C)c(C)c1OCC(=O)N(CC(O)CNC(=O)CC1OCCO1)C N1(C(=O)NCCOCCC#C)CC(C)c2ncccc21 C1(O)(C(=O)NC(C=C)C)CCN(C(C2(c3cccs3)CCCCC2)=O)CC1 Cc1ccc(CCC(=O)NC2(CNC(=O)Cn3cc(CN(C)C)nn3)CC2)s1 C1(NC(c2nccc(CC)c2)=O)CN(C(C2CC(=O)NC2(C)C)=O)CC1(C)C c1(C(C(=O)NC(CC)(C)C)N(C(c2cccnc2)C(=O)NC)C)ccc(I)cc1 C1(NC(C=CC(=O)OC(C)C(=O)c2ccco2)=O)CCCC(F)(F)C1 Cc1cccc(C(C)C(N2CC(n3cc(-c4ccns4)nn3)(C(=O)O)C2)=O)c1 C1(N(C(CC(CC)O)=O)C)CC2CCC(C1)N2C(c1ccc(F)cc1)=O c1(OC)cc(C(=O)N(C)CC2(O)CCCN(C(=O)CCSC)C2)ccc1C#N C(CCCC(=O)N(C(C)CN(C(=O)C(C)C#N)C)C)OC N1(C(CCN(C(=O)CCC2CC2(F)F)C(C)C)=O)CCOCC(C2CC2)C1 C1(CC(=O)NCC(CC(=O)N2CC(SCC)C2)C)CC2(CCO1)CC2 N1(C(C2(C)N(C)CCC2)=O)CCCC2CN(C(=O)C=C3CCCC3)CCC12 C(=O)(CCCCCC(C)O)NCCCN(C(c1ccc(=NC)[nH]c1)=O)C c1(CC(=O)N(CC(C)NC(c2c[nH]nc2OCC(F)F)=O)CC)nnc(S)n1C C(CCCCCNC(c1n[nH]c(C)c1Br)=O)NC(C(C)(C)OC(C)=O)=O N1(Cc2nnc(C(C)C)o2)CCCC(CO)(NC(=O)CC2CCC(C(N)=O)O2)C1 c1(C(=O)NC(CNC(C2(CC)COC2)=O)C2CC2)ccncc1C(F)F C1(COC)CN(C(=O)CC(Cl)Cl)CCN1C(=O)CCCOC(C)(C)C c1(OC)ccc(Cl)c(C(=O)NNC(C2C=CCN(CF)C2)=O)n1.C(C)(C)(C)NC(=O)O C(=O)(C(C)C(F)(F)C(F)F)NCC(CC=C)CO.c12ccccc1O2 c1(OC)cc(OC)c(C(N2CCC(NC(=O)CCNC(=O)C=CCl)C2)=O)c(F)c1 O=C(N=c1ccn(Cc2cccnc2)[nH]1)Nc1ncnc2sccc12 c1(C(N2CC3(N(C(C(CCCC)O)=O)CC3)C2)=O)cc2ccccn2n1 N1(C(CN(C(C)C)C)=O)CC(N(C)C(c2cc(Cl)nnc2O)=O)C2(CC2)C1 CC(O)(C(=O)NCCn1cnc(C(N2C3CSCC2C3)=O)c1)C(F)(F)F c1(OC)ncc(CNC(N2CCC(Nc3ncccn3)C2)=O)cc1C c1(C(N2CCC(NC(C3(CC#C)CCCC3)=O)C(F)C2)=O)cccc(C#N)c1C n1(CC(N2CCCC3(CNC(CCC)=O)C2C3)=O)nc2ccccn2c1=O c1(OC)cc(C)sc1C(=O)NCc1ccc(C(C)NC(=O)CC(C)F)cc1 C(=O)(CC(C1CC1)NC(C1(O)CCC1)=O)N(CC=C)CC1CC1 C1(CNC(C2(CCC=C)CN(C(c3ncn(C(C)C)n3)=O)C2)=O)CCOCC1C C1(NC(c2cccs2)=O)CC2CC1CN(C(c1cccc(OC(F)(F)F)n1)=O)C2 c1(C(=O)NC2C(C)CN(C(=O)CCC3CCCCC3)C2)ccn2cccc2c1 CC1CC(CNC(c2occc2CNC(=O)C2=CCCSC2)=O)CC(C)C1 C1(NC(=O)C(C(CC)N(C)Cc2cccc(OC)c2)OC)CS(=O)(=O)CC1O C1(C(=O)NCCOC2CN(C(c3cc(N)c(Cl)nc3)=O)C2)CCn2ncnc2C1 C(C)(CC(=O)NCC(C)C(=O)NC)N(C(C1C(C(=O)OC)C1)=O)C CCCCCC(O)C(=O)NCC1CCN1C(=O)C=Cc1cscn1 c1(C(=O)NCCC(C)Nc2ncnc(Cl)c2Br)cnc2[nH]c(O)nc2c1 c1(C(N2C(CNC(c3c(C)ccc(C)n3)=O)CC3CC32)=O)cn2c(n1)CCCC2 C1(N(C(CCC)=O)CC2CCCO2)CCN(C(=O)CCC2CCCN2C)CC1 Cc1cn2cc(CC(=O)Nc3cn(CC4CCOCC4)nc3C)nc2s1 C12(NC(=O)CCc3ccc(O)nc3)CCN(C(C3CCC=CCC3)=O)CC1C2 Cc1cc(C(=O)OCCC(=O)NCc2cccc(OC(C)C)c2)cc(O)c1 C(CCC(=O)N(C)Cc1ncc(COC)s1)NC(=O)OCC N1(C(c2c(=O)ccn(C)c2)=O)CCC2CN(C(=O)CSCC3CCCO3)C2C1 c1(CN(CC(O)CN(C(=O)CCCCOC(C)(C)C)C)CC)cccc(C#N)c1 N1(C(c2c(OC)c[nH]n2)=O)CCC(NC(c2cc(Cl)cc(Cl)c2)=O)CC1C Cc1ccc(C(=O)N(CCCCN(C)C(C2CC23CC3)=O)C)c(O)c1 c1(CC)cc(C(=O)NCC(C(C)(C)C)NC(C2CC3CCC3C2)=O)cc(N)c1 Cc1cc(C(=O)NCC(F)CNC(=O)Cc2c(C)noc2C)ncc1N c1(C2(CNC(c3n(C(CC)C)nnn3)C3CCC3)CC2)ccc(Br)c(Cl)c1 CC1CS(=O)CCN1C(C1CC2CCC1N2C(c1ncccc1Cl)=O)=O C1(C)(CNC(CC(C)(C)OC)=O)CCN(C(c2ccc(F)s2)=O)CC1 C1(C(=O)NC2(C)CC(NC(=O)Cc3cnc[nH]3)C2)COCCN1C=O N1(C(c2c(CCC)n(C3CCCC3)nc2)=O)CCC(COCC)C1(C)C C1(C(N2C3CC(CC(NC(C(C)(C)F)=O)C3)C2)=O)CCCCC12OCCO2 Cn1ncc2cc(C(=O)Nc3cccc(NC(c4ncnc(O)c4F)=O)c3)sc12 N#Cc1ncccc1-c1cn(CC2CCCN2C(c2ncccc2F)=O)nn1 c1(C2(C)CNC2)cn(CC(=O)NC2CC(n3cnnc3)C2)nn1 N1(CC(N2C(c3[nH]c(C(C)=O)c(C)n3)CCC2)=O)Cc2ccc(Br)cc2C1=O n1(CC(=O)NC(C)CCCNC(c2cccc(F)c2O)=O)cc(S(C)(=O)=O)cn1 C(=O)(C(C(CC)CC)OC)NCC(C(=O)NCC1CCC(CC)O1)(C)C C1(C(CNC(C(C)SCCCC)=O)O)CCN(C(c2cncn2C)=O)CC1 N1(C(C(C=CCCC)O)=O)CC(CNC(=O)CCc2cn[nH]c2)OC2(CCC2)C1 CCC(O)CCN=c1nc(OC)[nH]c(N(CC(C)OC(C)(C)C)C)n1 N1(C(c2sc(C)c(O)n2)=O)CCC(NC(=O)Cc2cccnc2Cl)C(C)C1 c1(CN2CCC(OC)(CN(C)C)CC2)cnc2ccccc2c1 c1(C(=O)NC(C(=O)NCC(C)OCC=C)Cn2cncn2)cc[nH]c(=NC)c1 N1(C(C=Cc2cn(C)nn2)=O)CCC(NC(=O)CCc2ccoc2)C12CCC2 N1(C(C(C)CO)=O)CCC2C(C(N3CCCC3(C)C3CCC3)=O)C2C1 CCC(C)CC(C)N(C)C(c1occc1CNC(C1(C(C)C)COC1)=O)=O c1(C(N(CC(C)N(C(=O)C(F)C(F)(F)F)C)C)=O)cccc(F)c1F C(=O)(C1c2ccccc2C2CC1C2)NCC1C(NC(c2nc(C(C)=O)sc2)=O)C1 C1(C(=O)OCC)CCCN(C(=O)Nc2cnn(C(C)(C)C)c2CN2CCCC2)C1 O=S(=O)(c1cc(Br)c(Cl)s1)N1CCC(Nc2cccc(Cl)c2)CC1 n1(CC)c(N)c(C(=O)Cc2cc(C)n(-c3cccc(C#N)c3)c2C)c(O)nc1=O c1(NC(C(CC2(C)CCOC2)N(CC(C(C)(C)C)F)C)=O)ccc2c(c1)OCO2 N1(C(CNC(C)=O)=O)CC2CC1(C(=O)NOCC1CC13CCC3)C2 N1(C(c2cc(Br)cs2)=O)CCC(F)(CNC(C2CC(F)C2)=O)C1 c1(C(N2CCCC(c3nccs3)C2)C(=O)NCC)cccc2cnn(C)c12 c1(NC(C(c2ccc(C)cc2)C)=O)nc2ccccc2s1.C12CC(C1)C(=O)N2 C1(CNC(=O)CCCc2cc[nH]n2)COCCN(C(c2cnco2)=O)C1 CCC(C)CC(=O)NCC1(NC(=O)CCc2ccc(SC)cc2)CCOC1 N1(C(C(CCC)(C)C)=O)CC2CCCC(NC(C3CCSC3)=O)(C2)C1 C1(N(C(=O)CCCc2ncco2)CC)CCCN(C(C2(F)CC=CC2)=O)C1 c1(SC)ncc(N)c(C(=O)N(CCC(F)(F)F)C(C)C2CC2)n1 C1(C(N(CC)CC2CC2(F)F)=O)CCCN(C(=O)C(F)CC2CCOC2)C1 C(C)(CCCCC#N)(c1nnnn1CSc1ccccc1)NCC(CCC)OC N1(S(C(C)C)(=O)=O)CCC2(CC2C(=O)Nc2ncc(Br)nn2)C1 c1(C(=O)NC2CCC(NC(c3ccns3)=O)C2)ccc(F)c(Br)c1 c1(C(N2CC3C(NC(CCC4N(C)CCC4)=O)C3C2)=O)c(F)cccc1[N+](=O)[O-] c1(C(=O)NCC(CNC(CN(C)C(N)=O)=O)O)cc(C2CCCO2)n(C)n1 N1(C(C(CC)Oc2ccc(C)cc2C)=O)CCC2(CC1)CNCC2C(=O)O c1(C(=O)NC2CC(OC)CN(C(C3CCOC3)=O)C2)cc2ccccc2n1C c1(C(N(CC(=O)NC(C)(C)CO)CC#C)=O)cscc1OC C1(CN(C(CCN(C(=O)C(C)=C(C)CC)CC=C)=O)C)CCCCO1 N1(C(C(C2CCC2)OC)=O)CC(NC(c2nocc2C(C)C)=O)C2CCCC2C1 c1(C(=O)NC(C(C)C)CNC(C2CN(C)C(=O)N2)=O)cccc(C#CC2CC2)c1 CC(CCCNC(=O)CCC1CCOC1)NC(=O)C(C)Sc1ccccc1 c1(C(N2CCC(C)C(NC(c3ncccc3F)=O)C2)=O)ccc(Cl)c(C#N)n1 CC(C)CC(F)(F)C(=O)NC1CCCC(NC(c2ccc(F)c(F)c2)=O)CC1 c1(OC)cc(C(N2CC(C)C(C)C2)=O)c(-c2cnc(=N)[nH]c2)cn1 CC(C)CS(=O)(=O)CC(=O)N1CCN(C(C2CCC(=O)N2C)=O)C(CC2CC2)C1 C1(C(N2CCCC(CCCC)C2)=O)COC2(C1)CN(C(c1c[nH]c(=O)cn1)=O)C2 C1(NC(C(C)OCCC#C)=O)CN(CCOc2ccccc2OC)CCC1C N1(C(CN(c2ccccc2)C)=O)CC(C)(C)OCC1CNC(=O)C1=CCCSC1 c1(CC(=O)NC(CNC(C=CC)=O)CCOC)cc(Cl)c2c(c1)OCCO2 c1(C(N(CC(CC)NC(C2CNC(=O)C2)=O)CC)=O)n[nH]c2ccc(OC)nc12 C(=O)(CC(C)(CN(C)C)C(F)(F)F)NC1C2CN(C(COCCCCC)=O)CC21 N1(C(CN(C(C(C=CC)O)=O)C2CC2)=O)CCCC2(CC(O)C2)C1 C1(C(N2CCC(N(C)C(c3n[nH]cc3Br)=O)CC2)=O)CCn2nnnc2C1 c1(C(=O)NCC(C)(CC)NC(CCCCC)=O)cc2ccccc2c(O)n1 C(=O)(C(C)CC(C)(C)C)NC1C(n2cc(CCCSC)nn2)CCCC1 C1(c2c(COC(C3C(C(C)C)OCC3)=O)cnn2C)CC2(CCO1)CC2 C1(C)(C(N2CC(CNC(c3nc(CC(C)C)sc3)=O)C(C)C2)=O)CCC(O)CC1 C1(C(C)C)CN(C(=O)CN(C)C)CCCN1C(=O)CSCc1nccn1C c12ccc(cc1)CC(=O)N(C1CC1)C2.C1(C(=O)NC2C(CC)C2)CCCN1CC CC(C)C(C)C(=O)NC1CCCC1CNC(=O)CCNC(=O)NCCCO N12CC(OC)C(C1)C2=O.C(=O)(CS(C)(=O)=O)NC1N(CCC)CCC1 C1(NC(C2(C)C=CCC2)=O)CCCC2CN(C(c3nc(C(C)(C)C)no3)=O)CC12 C#Cc1cccc(C(c2nnnn2C2(C)CC2)NCc2nn(C)cc2C)c1 C12(CNC(C)=O)COCCN1CCN(C(C1CCC3CCC1O3)=O)C2 Cc1cc(C(N2CC(C3CN(C(=O)C=CBr)C3)C2)=O)c2[nH]cnc2c1 C(=O)(C(C)(C)S(C)(=O)=O)N1C(CNC(c2ccc(C(C)C)cn2)=O)C2CCC1C2 C(c1ccco1)=C(C)C(=O)NCCCOCCOCCNC(C1CCSCC1)=O CC(CO)N(C)NC(=O)C1(C)CCNC(=O)CC1 N1(C(C2(SC)CC2)=O)CCCN(CCCCNC(C2(C)CC(F)(F)C2)=O)CC1 c1(CNC(C2CCC2c2nnc(S)o2)=O)cnc2ccccn2c1=O CON1CCC(CC(N2CC(N(C)C(c3cnnc(O)c3)=O)C(O)C2)=O)CC1 C(=O)(CC(=O)NCC1CC(NC(=O)CCC2CC2CC2CC2)C1)OC CCCCCCC(F)C(=O)NC1(CNC(c2ccc(C(F)(F)F)o2)=O)CCC1 c1(C(N2CC(C(C)(C)O)(CNC(C(CC)O)=O)C2)=O)nnn(C)c1COC c1(CC)ncoc1C(N1CC(CO)(NC(c2cnn(CC3CCOC3)c2)=O)C1)=O N1(C(C(COC)OC)=O)CC(NC(=O)C(=Cc2cccnc2)C)C(C)(C)C1 C(=O)(C1CCCc2cccnc21)NCCCC(C)NC(c1c(CC)oc(C)c1)=O CC1=NOC(CC(=O)NCCOCCC(=O)NCc2ccncc2)C1 N1(C(c2ccc(OC)cc2N)=O)CCCN(C(C2C(C)C2C)=O)CC1C N1(C(C(C)S)=O)CC2CCN(C(c3c(Cl)ccc(Br)c3F)=O)C2C1 N1(C(c2c(CC)nn[nH]2)=O)CCCC(CNC(=O)CC2CNC(=O)C2)C1 Cc1cc(C)c(C(=O)N(C2(C(N3CC(CO)CC(C)C3)=O)CC2)C)cn1 N12CCC(C(F)(F)C1)C2.c1(SC)nccc(NC(c2cnc(C3CC3)nc2)=O)n1 C(=O)(CCCCC(C)(C)C)N1CC(NC(COC(CC)(C)C)=O)N(C)CC1 C1(NC(C2CC3(C2)CC32CC2)=O)CC2CCC(C1)N2C(C1C2(CC2)C12CC2)=O C1(C(=O)NC2(CC)CCOC2)CN(C(=O)C2=C(C)CCC2)CC(C)(C)C1 CCCC(C)CC(=O)NCC(CC)N(C(=O)CC1COCCN1CC)C C(=O)(C(C)C(F)(F)C(F)F)NC1C2(CN(C(c3n(CCC)nc(C)c3)=O)C2)CC1 Cc1ccc(C(C)CC(=O)N(CCC(C(C)C)NC(c2csnc2C)=O)C)cc1 N1(C(c2cnc(CC)[nH]2)=O)CC(NC(c2c(Cl)n[nH]c2C)=O)C(C)C1 C=CCCC(F)(F)C(=O)NCC(O)CCNC(=O)CCc1cc(OC)no1 CC1(C)CC(NC(c2cnc(O)s2)=O)CN1C(=O)CC(=O)NCC(F)(F)F c1(C(N2CC(C)(CNC(CSC)=O)OCC2)=O)cnc2snc(C)c2c1 N1(C(COCCOC)=O)CCC(CC(=O)NCCC(=O)NC(N)=O)C1 C1(N(C)C)(C(N2CCCC2CNC(=O)CCC2CCC2)=O)CCCSC1 C1(NC(C2C(C)(C)CO2)=O)(CNC(=O)C=CC2CCCCC2)CCC(F)(F)CC1 C1(CNC(C(COCC)C)=O)(NC(c2sc(F)cc2Cl)=O)CC2CCC1CC2 N1(C(c2n(C=C)ncc2)=O)CCN(C(=O)CCc2cnc(C)s2)C2CCCCC12 C1(C)(C(=O)NCCC2CCN(C)C2)CN(C(C2CN3CCN2CC3)=O)C(C)(C)C1 C(=O)(C(CCOCCO)NC(c1cc(C)oc1C)=O)NCC1N(CC)CCC1 C(=O)(CCN(OC)C(=O)C1CC2(CCN1C(=O)CCC1CCCO1)CC2)OC C1(C(C)(C)CNC(=O)C(O)C2CCCC2)CCN(C(c2sccc2CO)=O)CC1 C1(CC=C)(NC(c2[nH]ccc2CNC(C2C(C(C)=O)C2(C)C)=O)=O)CCCC1 C1(NC(c2cc(C)c(C)s2)=O)CC2CC(NC(c3ccnc(O)c3)=O)C1C2 S(=O)(=O)(c1cn[nH]c1)NC(COC1C(C)CCCC1)=O C(C(C)NC(c1ccnn1CC1CC1)=O)(C(C)C)NC(COCCCC)=O C1(NC(C2(C)C(CC)CCC2)=O)COC2(C1)CN(C(C1CC3C=CC1C3)=O)C2 c1(NCC2=C(Cl)C(S(C)(=O)=O)=C2)cc(=NC2CCC2)[nH]c(C(F)(F)F)n1 C(C1c2ccccc2CCN1C(=O)C=CC1CCCC1)NC(c1coc(O)n1)=O N1(C(C(c2ccn(C)n2)C)=O)CCN(C(=O)C(C)CC2CCCC2)C(C2CC2)C1 c1(CCC(=O)NCCN(C(=O)Cn2cc(C#N)cn2)C)c(F)cccc1F CCCCC(C(=O)Nc1cn(CCF)nc1C)NC(c1cc[n+]([O-])cc1)=O c1(C(=O)NCC2CCC(C)CN2C(=O)CCOC2CCC2)c(Cl)ccc(F)c1N c1(C(=O)NC(CN(C)C)C(=O)NCCCC2CCOC2)ccccc1O C1(CC)(NC(c2nccn2C)=O)CCCN(C(C2CC(=C(F)F)C2)=O)C1 N1(C(c2c(C)nco2)=O)CC=CCC1C(=O)NC(c1cccc(F)c1)C c1(C(N2CCN(C(C3CN(C)C3)=O)CC(CO)C2)=O)cccc2cc(Cl)ccc12 c1(C(N2CCC(N(C(C(CC)OC)=O)CCO)C2)=O)ccc2ccn(C)c2c1 C(=O)(CCC(CF)CF)N(CCN(C(=O)CC1COCC1(C)C)C(C)C)C O=S(=O)(c1ccc(Br)cc1N1CCn2cnnc2C1)NC1CCCC(F)C1 C1(C(N2CCCC(C)C2)=O)CCN(C(C2CC23CCCCC3)=O)C12CC2 c1(CNC(=O)CC2N(S(CCOC(C)(C)C)(=O)=O)CCC2)ccc(Br)cc1 c1(C(N2CCC(F)(CNC(c3coc(C4CC4)n3)=O)C2)=O)cnc2[nH]cnc2c1 c1(-n2cc(C(CC)(O)CC)nn2)cc(C(N2CC(C(=O)N(C)C)C2)=O)ccc1C C=CCC(C(=O)N1CC=CC1CNC(=O)CC1CCCC12CC2)NC(C)=O c1(OC)c(Br)cc(C(N2CC3CN(C(c4csc(C)n4)=O)C3C2)=O)cc1Br N1(c2ccc(C(=O)OC(C)(C)C)cn2)CC2CCCC2(C(N)=O)C1.c1(=O)c(=O)[nH]1 CC1C(NC(=O)COC2COC2)C(C)CCN1C(=O)CCc1ccn(C)c1 c1(NC(C2(SC)CN(C(=O)C(F)CCC(C)C)C2)=O)ccc(C)c(O)c1C c1(CC)ccc(C)nc1NC(C1C=CCN1Cc1nc(-c2ccccc2)cs1)=O C12(CNC(c3cccc(F)c3F)=O)CCCCC1N(CC#N)CC2 Cc1ncc(CCC(=O)NC(CN(C)C)C(=O)N2CC(O)(CN(C)C)C2)o1 N1(C(c2c(C)noc2C(F)F)=O)CC2CCC(NC(=O)CC3CC3(Cl)Cl)CC2C1 N1(C(C2(CC)CCOC2)=O)CC(N(C(=O)CSCCC#N)C)C2(CC2)C1 C1(NC(CC2C3CN(C(C#CC(C)(C)O)=O)CC32)=O)CCCCCCC1O N1(C(CC2C(=O)NC(=O)N2)=O)CCOC2CN(C(C3CCCS3(=O)=O)=O)CC12 C(=O)(CC(C1CC1)NC(=O)C(C)(O)C1CCCCC1)NC c1(N(CC(F)Cl)C)ccc(S(=O)(=O)NC2(CO)CCOC2)c(Br)c1 C1(C(=O)NC2COC3CN(C(C4C(C#C)C4)=O)CC32)C2CC3CC(C2)CC1C3 C(C(=O)Nc1ccc(S(=O)(=O)CC2CCCCC2)cc1)(C(C)C)(C(C)C)NC(C)=O N1(C(c2c(C)oc(C#N)c2)=O)CCC2(CC1)CN(C(c1cc(Cl)cc(Cl)c1)=O)C2 C1(CCNC(C=CSC)=O)CCN(C(=O)C(F)=C(C)C2CC2)CC1 C1(NC(Cc2cn(CC)nc2)=O)CCCCC1CNC(=O)C(CO)OC C1(C(N2CCC(n3cnnn3)C2)C(=O)NCCOC)CCC(SC)C1 Cc1c(C(=O)NC2CC(NCCCC(=O)CSc3cccc(F)c3)C2)nn(C)c1N C1(CC(=O)NCCNC(c2c(OC)ccc(C(N)=O)c2)=O)CCCCCC1(F)F N1(CC)CCOC(C(=O)N(CCNC(C2(C)CC2(C)C)=O)C(C)C)C1 c1(C(=O)Nc2cc(O)ncn2)ccc(S(=O)(=O)N2CCCCC2)cc1 Cc1oc(=NC2CC(n3ccnn3)C2)[nH]c1C(=O)OCC(N1CCCC1)=O N1(C(C=CCC)=O)CC2(CNC(C3(OCCOC)CCOC3)=O)CC(F)(C1)C2 CC1(C)CCC(CC(N2CCCC2C(C)(C)NC(=O)C2CC2)=O)OC1 C1(CC=C)(NC(=O)Cc2cnnn2C)CCN(C(=O)C(F)C2CCC2)C1 c1(C(N2CC(F)(CNC(C3(C)CCC(C)C3)=O)C2)=O)cc2n(n1)CCNS2(=O)=O N1(C(C(CCOCCO)NC(CCCC)=O)=O)CC(O)(C2CCC2)C1 Cc1ccc(NC(=O)N(C)C)c(C(=O)NCCC(C)N(C(=O)C(O)C(F)F)C)c1 c1(NC(=O)CN2CCCC2C(=O)CCc2ccccc2)ccccc1Br N1(C(COC(C)=O)=O)CC2CC(NC(c3cnc(C(F)F)nc3)=O)CC1C2 C(C(CC(=O)NC1(CO)CCNC1=O)NC(C1CC=CC1)=O)OC C1(NC(COC(C)(C)C)=O)CCCC1C(=O)Nc1ccnn1C1CC1 N=c1[nH]c(CCC(=O)NCCNC(c2sccc2OC(F)F)=O)cs1 N1(C(c2c(C#N)csc2)=O)CC(C2(NC(=O)Cc3cncs3)CC2)C1 CCC(CC)(CO)C(=O)NCCC1CCN(C(c2ccc(=N)[nH]c2OC)=O)CC1 C(CC1c2ccccc2CCN1C(=O)C(F)=C1CCC1)NC(=O)CC1CCCC1 N1(C(C2(SCC)CC2)=O)CCC(O)(CNC(=O)C(C(C)C)NC(N)=O)C1 N1(C(C(CC)n2ccnc2)=O)CC2(CC(C(=O)NC(COC)C(=O)OC)CO2)C1 C1(CCNC(=O)Cc2cscn2)(C(N2CC(n3ccnn3)C2)=O)CCCC1 C#CCC(C(=O)N(C(C)C(C)SC)C)NC(=O)C=C(C)C1CC1 C1(c2nc(C(c3ccc(N4CCCS4(=O)=O)cc3)C)on2)CCc2nn[nH]c2C1 c1(CC(=O)NC(CCNC(C(CC)(C)F)=O)C(C)C)ccc(Cl)cc1F c1(CNCc2ccc(C(N)=O)s2)ccc(Br)cc1I O(C1CCCc2ccccc21)CC(=O)NC1CCC(NC(C2CCSCC2)=O)C1 N#Cc1cc(C(=O)OC2CCC(C#N)C2)cnc1C(F)(F)F c1(C2C(C(=O)NC(C3CCN(C(c4cnco4)=O)C3)C)C2)cccnc1 c1(C(=O)NC2(CC(=O)N(C)CCn3cccn3)CC2)ccncc1 CCC(C)CCC(=O)NCC(C)CNC(=O)COc1ccccc1C N1(C(CNC(CC(C)(C)C)=O)=O)CCN(C(=O)C(C)(C)C(N)=O)CC(C)(C)C1 N12CCCCC(C1)CCC2=O.O=C(CC(=O)N1CCCC1CO)NC1CC1 N1(C(c2c(C)c[nH]n2)=O)CC(CNC(C2C3CNC(=O)C23)=O)C(C)(C)C1 C#CCC(C)C(=O)N(C(C)CNC(c1ccc(NCc2ccco2)cc1)=O)C C(=O)(C(F)(F)C(O)C(C)C)NC(CCNC(C1(CCOCC)CCC1)=O)(C)C C1(C(CNC(c2cc(OC)ns2)=O)(C)O)CCN(C(C2CCC(=O)O2)=O)CC1 c1(C(N2CC(C(C)NC(C=CC=CC)=O)C2)=O)cc(O)cc(C#N)c1 C(=O)(C(CC(=C)C)OC)N1CC(C(=O)NC(c2ncc[nH]2)C#C)(CC)C1 n1(CCCC)ncc(C(=O)NC2CC(O)(CNC(C3CC=CCC3)=O)C2)c1C C1(CNC(COCCCC)=O)CN(C(=O)C(C)CC(F)F)CCC1(C)C C1(NC(CSCc2cccc(C)c2)=O)CN(C(c2nc(C)no2)=O)CC2(CC2)C1 c1(C(=O)NCCOCCCF)ncccc1Cl C(=O)(C(F)C(C)(C)O)NC(CC=CC)C(=O)N1CC(CO)C1(C)C C(=O)(CCC(F)(F)F)N(CCC)CCNC(C1(C)CC2CC2C1)=O c1(COC)nc(CC(=O)NC(C2CCN(C(C3(n4cncn4)CC3)=O)C2)C)cs1 C(CC(C(=O)N1CCNC(=O)C1)NC(=O)CC1CC(C2CC2)C1)N(C)C c1(CN2CCC(NC(c3c(SCC)cccc3)=O)C2)c(Cl)cccc1I N1(S(CCC(C)(C)C#N)(=O)=O)CC=C(c2cccc(Br)c2)CC1 C12(Cn3cc(C4CCC(NC(C5(SC)CC(C)C5)=O)C4)nn3)CC(C1)C(C)(C)O2 c1(C(N2CC(CNC(C3(C(F)(F)F)CCN(C)C3)=O)C(O)C2)=O)cccc(F)c1F CCC(C)(CNC(=O)C(C)Cn1cccn1)C(=O)NCCC1CCC(C)(C)O1 c1(CCC(N2CC(COC)(NC(c3cc(Cl)n(C)n3)=O)C2)=O)cnc(C)nc1O C1(NC(C(C)C(C)O)=O)C(C)(C)CN(C(=O)CCC(N)=O)CC1(C)C CC1CCC(CO)N1Cc1ccns1 C1(C(=O)NCC(C)CC2CC2)COCC1NC(C1CC1Cl)=O CCCC(C#N)C(=O)N1CC(O)CC1CNC(=O)CCc1nnc(O)nc1O CCCCC(C)(F)C(=O)NCC(c1ccc(N(C)C)cc1)NC(C1CC2CC2C1)=O C(=O)(C1=Cc2ccccc2C1)NC1CCN(C(CC2ON=C(C)C2)=O)C(C)C1 N1(C(C(C)(C)OC)=O)CCN(C(C2(C)CCN(C(c3ccccc3)=O)C2)=O)CC1 C1(C(=O)OC)CN(C(=O)CCC2CCC(=O)N2)CC2(CCC2)O1 N1(C(C2CCC(C(=O)OCC)C2)=O)CC(C(=O)O)CC12CCOCC2 C1(C(=O)NC(c2cn(CC)nc2)C)CN(C(=O)CC2CSCCO2)C(C)(C)C1 c1(C(N2CC3C(CNC(C4CCC(OC)CC4)=O)(C3)C2)=O)cc2ccncc2[nH]1 Cc1c(C(=O)NC2(C)CCN(C(=O)CC3COCC3(C)C)CC2)nn(C)c1N c1(C(=O)NC2CCN(C(CNC(=O)OC)=O)CC2C)nccn2c(C)nnc12 Cc1ccc(=N)[nH]c1C(=O)NCC(C1CCCC1)NC(=O)CCN1CCCCC1C C1(C(=O)NCCC2CCN(C(c3c(C(C)C)con3)=O)C2)CSCC(=O)N1 C=CCCCC(C(=O)NCC1CCC(C)C1)NC(c1ncc(C)cc1F)=O c1(SC)ccc(C(N2CCCC2CNC(C2(N3CCOCC3)CCCC2)=O)=O)o1 N1(C(=O)NCCCl)CCC2C1CCN2C(c1ccc2n[nH]cc2c1)=O C1(NC(CCc2cc(C)no2)=O)CCN(C(=O)Cn2nccc2C)C12CCCC2 C12(C(=O)NCC3CN(C(=O)Cn4ccc(C5CC5)n4)CCO3)CCC(CC1)CC2 C=C1CCC(C(=O)NCCC(O)CNC(c2cccc(C(F)F)c2)=O)CC1 c1(C(N2CCN(CC(CC)CC)CC2)=O)cc2c(C)cccc2o1 C(=O)(CCC(C)(C)C#N)N1CC(CC(C)NC(CC(CC)CN(C)C)=O)C1 CCC(C)CC(C(=O)NCCOCCCF)NC(=O)C(C1CC1)SC c1(C(C(=O)NCCOC)N(CCOCC)C)ccnc(OC2(C)CCCC2)c1 C1(C(=O)NCC(CNC(c2cc(CC)[nH]n2)=O)OC)CCc2c(nnn2CC)C1 N1(C(C=Cc2c(C)nccc2)=O)CCN(C(c2cc(CO)[nH]n2)=O)C(C)C1C c1(C(C(=O)NCC2(CNC(C3CCC(C)C3)=O)CC2)=O)ccc(Cl)cc1 C1(CC(=O)NC2(COC)CCC2)CCN(C(C2C=C(C)CS2)=O)C1 C(=O)(CS(=O)(=O)C1CC1)N1C(COC)(CNC(=O)CC2C(C)C2(F)F)CCC1 c1(C(=O)NCC2CCC(C(N(C3C(C)CCC3)C)=O)O2)ccc(C#N)s1 Cc1nn(CCC(N2CC(CNC(c3cncnc3)=O)CC2C)=O)cc1Br c1(C(N2CCC(N(C(c3c(C)scc3)=O)C)C2)=O)cc(O)c2nc(C)n(C)c2c1 C=Cn1nncc1C(=O)N(C(C)C(=O)Nc1csc(Cl)c1)C1CC1 C1(N(C(CSCC)=O)C)CCCN(C(=O)CN2CCCCC2)CC1 N1(C(=O)NCCC#CCO)CC(CNC(=O)C(F)(F)F)C(c2ccccc2)C1 N1(C(CC=CC=C)=O)CCC(C(C)C(=O)NCCS(C)(=O)=O)CC1 C#Cc1cccc(C(=O)NC2CN(C(c3cnnn3C)=O)CC2O)c1F c1(CC(=O)NCC(CC)(C)NC(c2ccc(C(F)F)cc2)=O)ccc(Cl)nc1 c1(C(N2CCN(C(CCC(C)OC)=O)CC2)C(=O)O)ccc(F)c(Cl)c1 CC(C)CCC(F)C(=O)N1CC(CNC(=O)C=Cc2cscn2)OC(C)(C)C1 c1(CCNC(N(CCOCC=C)C)=O)cnn(C)c1 CC1OCCC1CC(=O)NCCn1cc(CNC(C2CC23CC3)=O)nn1 C(=O)(C(C)C(C)NC(C1CCCCC1)=O)NCC1C(OCC)CC1 C1(C(=O)NC(c2c(C)cccn2)c2ccccc2)(N(C)C)CCCCCC1 C1(NC(C2CSCCN2C(=O)CCCC2CC2)=O)CC12CC(O)C2 C(CN=C(NC1CCOCC1)NC1CCNC(=O)C1)N1CCC(C)CC1 CCC(CN(C(=O)COCC1CCC1)CC)NC(=O)C(C)SC(F)(F)F C=CC1OCCC1C(=O)NCCCCCCN(C(=O)C(F)C1CCC1)C C1(c2nnnn2CCC2CC2)(NCC(c2scc(C)n2)C)COCCOC1 N1(C(CCC(C)(C)F)=O)CCC2(COC(CNC(=O)CCCCCF)C2)C1 N1(C(CC(C(C)C)C)=O)CC(NC(c2ccc(CO)cc2F)=O)CC(C)(C)C1 N1(C(CC)=O)CCN(C(=O)C=CC2CCCN2C(=O)CC(F)(F)F)CC1 c1(CN(CCCNC(C(C)O)=O)C(c2ccoc2C(F)(F)F)=O)cccnc1 C1(NC(c2cc(C(N)=O)ncc2)=O)(CO)CCCN(C(c2cncc(F)n2)=O)C1 N1(C(C2COCCN(C(C3CCN(CC)CC3)=O)C2)=O)CC2CCN(C)CC2C1 N1(C(CC2(C)CC(F)(F)C2)=O)CCC(NC(=O)CC2CCC2)CC1C1CC1 Cc1cc(C(N2CCOC(CNC(=O)CC3(O)COC(C)(C)C3)C2)=O)cnc1O Cc1ccc(C(N2CC3CC3C2C(=O)NCCn2ccnc2)=O)c(O)n1 c1(C(=O)NCC2(F)CC(NC(CCOCCOC)=O)C2)ccc(Cl)cc1C C(CC(C)CC)(C(=O)N(C1(CCO)CC1)C)NC(C(CC#C)O)=O C1(CNC(C(C2CCC2)OCC)=O)CCCCN1C(=O)CC(C)N(C)C C1(C(N(C2CC(CO)C2)C)=O)CC2(CC2)CN1C(=O)Cc1ccco1 C1(CNC(Cc2scc(C)n2)=O)CC(NC(=O)CCS(C)(=O)=O)C1(C)C c1(NCCC2(OC)CN(C(c3cnc(Cl)s3)=O)C2)[nH]c(=O)n(C)c(=O)c1C#N c1(C(=O)NCCN(C(=O)CSC)OCC)cc(C(N2CCCC2)=O)sn1 CC1(NC(=O)C(CNC(=O)COC2(C)CCCC2)CC2CC2)CS(=O)(=O)C1 c1(C(=O)NC2C(NC(c3cnc(CC)s3)=O)CCC2)noc(C)c1[N+](=O)[O-] N1(C(c2cccc(OCC)c2)=O)CC2CC(NC(c3ccsc3OC)=O)CC2C1 c1(C(=O)NC(c2cccc(C)c2)CNC(CCCSC)=O)ccc(Cl)c(F)c1N c1(C(=O)NC(C2CCN(C(CCS(C)=O)=O)C2)(C)C)cc(S(C)(=O)=O)co1 CN1CCC(C(=O)N(CCCNC(=O)C(C)(C)C2CCC2)C2CC2)C1=O N1(C(C2CCC(CNC(Cc3c(C)ccs3)=O)C2)=O)CCCC(C)C1 C1(C(N2CC(OC)(CNC(=O)CN(C3CCCC3)C)C2)=O)C(Cl)(Cl)C12CC2 C1(O)(CCNC(=O)C2=CCSC2)CCCN(C(=O)C(F)C2CCCC2)C1 C1(C(=O)NCC(=O)NC)CCN(C(C2CN(C)CCO2)=O)CCO1 c1(N(C)Cc2ccn(C)n2)nc(N2CCC(CS(C)(=O)=O)C2)nc2cccnc12 Cc1c[nH]c(CC(N)=O)c1C(=O)NCC1(NC(c2[nH]ncc2C#N)=O)CC1 N1(C(CC=CC=C)=O)Cc2ccccc2C(NC(=O)CN2CCC(F)(F)C2)C1 C(=O)(C1CCc2c[nH]nc21)NC(C1CN(C(=O)CCOCCN(C)C)CCO1)C N1(C(C2C(C)(C)C2NC(C2CCC(C3CC3)C2)=O)=O)CC2(C)COCC2(C)C1 C1(NC(=O)Nc2cccc(OCCOC)c2)CCCCCCC1OC c1(CCN=C(NC(C=C)C)NC(c2ccccc2)C)noc2ccccc12 c1(CC)nccnc1NC(c1cc(NC(c2cc(C)nn2C)=O)cn1C)=O CCC1=C(C(=O)NCC(C)(CO)NC(c2cc(COC)cn2C)=O)SCCO1 C1(C(=O)NCC2CC(NC(C3(C=C)CC3)=O)C2)CCC2C1C2(F)F N1(C(c2ncn(C)c2)=O)CC(NC(c2cscc2C(F)(F)F)=O)CC(O)C1 C1(NC(c2c(OC)nccc2)=O)CC2CCC1CN(C(=O)Cn1[nH]cnc1=N)C2 CC1OC2(C(N3CCC(CN(C)C(C4OCC5CCCC45)=O)C3)=O)CCC1CC2 CC(=O)CCCC(=O)NCC(C)(C)CC(=O)NCC12CCCCC1C2 c1(NC(COCC(=O)N(C)C)=O)cccc(C(=O)NC2CNC(=O)C2)c1 CCC(CC)C(F)C(=O)N1CCCC(N(C(c2[nH]cnc2C)=O)CC2CC2)C1 N1(C(c2cnc(C)nc2)=O)CCCC(CNC(=O)C(C)Cc2cnc[nH]2)CC1 c1(C(=O)NC(C)(CNC(=O)CCCC(F)F)CO)cc(O)nc2ccccc12 Cn1ncc2c(NCCC=CBr)[nH]c(=NCC3CCOCC34CCCC4)nc12 N12C(CC1C)NC(=O)C2=O.C(C)(CC(=O)NC)OCC C=CC(CCC)CC(=O)N(C)CC1CCN(C(c2oc(CC)cc2C)=O)C1 C1(C(=O)Nc2cncc(OC)c2)CC12CCN(C(=O)C(C)N1CCCC1)CC2 C1(C)(OC)CC2CC1CC2NCc1csc(C(C)(C)C)n1 Cc1cccc(OCC(=O)NCC2CC3(CC3)CN2C(C2CCCSS2)=O)c1C C1(C(=O)NC(CCCNC(c2c(C)c[nH]c2)=O)C)CC12CC(OC(C)(C)C)C2 Cc1nscc1CC(=O)N(CC(O)CNC(c1c[nH]nc1C(F)(F)F)=O)C C(=O)(C1CCc2nccn21)N1CCN(C(c2c(C)c(Br)cnc2)=O)C(CO)C1 c1(NC(C2C(NC(=O)Cc3ccccc3C(F)(F)F)C2)=O)cc(O)cc(O)c1 C(=O)(CC(CN(C)C)CC)N1CCC(N(C(C2CC(=C)C2)=O)C)C1 n1(CC)ccnc1C(c1nnnn1CCOC)NCCC(=O)N(C)C c1(C(=O)NC2C(F)CCN(C(CC3CCC(C)(C)C3)=O)C2)cc2n(n1)CCCO2 c1(CC)cc(C(=O)NC(C)CC2CN(C(C3CC(C)(CC)C3)=O)C2)ccn1 C1(NC(CCc2c(C)noc2C)=O)CS(=O)(=O)CC1NC(c1cn(C)cc1C)=O N1(C(C(C)CC(F)F)=O)CC2CN(C(=O)C(C)(C)C#N)CC(F)(F)C2C1 C1(CNC(c2cnc(C)nc2C2CC2)=O)CCC(C)(C)CN1C(C1CC1(Cl)Cl)=O C12(CCCCC1)C(=O)N2.C1(CNC(CNC(C)=O)=O)CN(C)CC1C(F)(F)F CC(C)CCC(O)C(=O)N1CCOCC1CNC(=O)Cn1ccnc1C(C)C CC1(C(N2CC(F)(CNC(=O)Cn3cc(C4CC4)cn3)C2)=O)CC2CC2C1 c1(CC(=O)NC(CCNC(C(C)(C2(C)CC2)OC)=O)C)c(C)noc1C n12nnnc1C(c1cnc(O)s1)NCCC2.C(CCCC)SC C(CC(C)C)(C(=O)NCC(O)CC(=O)NC)NC(C(C)OCCCC)=O CC(CC(F)(F)F)C(=O)NC1CC(C(F)F)(NC(=O)CCc2nncs2)C1 c1(C(N2CCCN(C(C(C(C)C)OC)=O)CC2)=O)cc(C)cc(Cl)c1N C1(NC(=O)CC2CCS(=O)(=O)C2)CN(C(C23CSC(C2)C3)=O)CC1C1CC1 c1(NC(Cn2cc(C(CC)(O)CC)nn2)=O)ccc2c(c1)CCO2 c1(C2CC(C(=O)NCC(CNC(Cc3c(C)ccs3)=O)C)C2)cccc(F)c1 c1(C(=O)NC2CCC(CCNC(C(C)(F)F)=O)C2)nncc2ccccc12 c1(C(c2nnnn2C2CC(F)(F)C2)NCCCOCCOC)csc(C(F)F)c1 CC(C)(O)C#Cc1ccc(CN(C=O)CC2CCC3(CCC3)C2O)cc1 C1(COC)CN(C(C2CC(F)C(=O)N2)=O)CCN1C(=O)C(=O)N(C)C c1(C(=O)NCCCCN(C(C(CC2CCC2)OC)=O)C)ccc2nccn2c1 C1(NC(C2(NC(C)C)CC2)=O)CC2CCCC(C1)N2C(C1CC(C)C1)=O c1(N2C(C)CC(NC(CCC(=O)NCC)=O)C2)nc(C(F)(F)F)ccc1C#N c1(C(N2CCC(NC(C(CCC)C)=O)C(F)C2)=O)ccc(F)c(C#N)c1 c1(CC)c(N2CCC(C)(NC(c3ccc([N+](=O)[O-])o3)=O)CC2)ncnc1Cl C(CCCC(=O)N(C1CCN(C(c2cncnc2C(C)(C)C)=O)C1)C)SC c1(C(=O)NC(Cn2cc(C(=C)C)nn2)C)cc2cc(Cl)ccc2n1C N1(C(C(CC)OCC)=O)CC=C(CNC(c2c(Br)nnn2C)=O)CC1 N1(Cc2ncc(C)nc2)CCN(c2ncc(C(F)(F)F)cn2)CC1C N(C(=NCCCF)NCC(C)(O)CC)C(C#C)CCC Cc1c(F)ccc(NC(C2CSC(=O)N2)=O)c1F C1(CC(N2CCC(N(CC)NC(=O)CC3(SC)CC3)C2)=O)CCCC12CC2 c1(C(=O)NCC2CC(F)(CNC(C3C(C#N)C3)=O)C2)ccc2snnc2c1 c1(OC)cncc(C(N2CCC(NC(=O)C3=CC(C)(C)C3)C2C(C)C)=O)c1C C1(C(=O)NC(c2cccc(C)c2C)C(=O)OC)CCC2OCCC2N1 C1(C(=O)NC2CC(CCF)C2)CC12CCN(C(=O)C(F)C(F)(F)F)CC2 C(=O)(CCS(C)=O)NCC(CC)(C)NC(=O)CCC(=O)c1ccc[nH]1 C(=O)(C(C)(F)C(F)(F)F)NC1C(C)CN(C(=O)CCn2cccnc2=O)C1 N1(CCC(N2C(C3(NC(C4CCC45CCC5)=O)CC3)CCC2)=O)CCCCC1=O C(C(O)CN(C)C(C1CCCC1)=O)N(C(=O)CCNC(c1cccs1)=O)C CCC(C)C(C(=O)NCC(=O)Nc1ccc(CCO)nc1)N(C)C C(=O)(CS(C)(=O)=O)N(C(CC)C(=O)NCc1coc(C)n1)C c1(-c2cc(C)cc(C)c2)ccc(S(=O)(=O)NCc2cnc3occc3c2)s1 N1(C(CC=CC=C)=O)CC(C)C(C)(CNC(c2nn(C)c(Br)c2C)=O)C1 C(=O)(C1=C(CCl)N(CC2CCCO2)C(=O)NC1c1ccc2ccoc2c1)OCC C1(F)(CNC(Cc2scc(C)c2)=O)CCCN(C(=O)C(N2CCCC(O)C2)C)C1 c1(C(N2C(CNC(c3c(C)cc(=N)[nH]c3)=O)CC2)=O)cc(C)c(Br)c(C)c1 C(C)(CC(C)CC)N(C(C1(NC(COCCCC)=O)CCCC1)=O)C N1(C(c2ccc(CC)s2)=O)CCN(C(c2ccc(F)c(C)c2)=O)CC1CO c1(CC)cn2c(n1)CCC(C(=O)Nc1cc(C(=O)OC)c(Br)c(C)c1)C2 C1(NC(C2N(C(C(c3cncnc3)C)=O)CCC2)=O)CN(C)CC1C C1(N(C(c2c(C)con2)=O)C)CCCN(C(=O)C=Cc2cn[nH]c2)C1 c1(CC)nn(C)c(N2CCN(C(=O)COCC(F)F)CC2CC)c1[N+](=O)[O-] c1(OC)cc(Cl)ccc1C(=O)NC(C)CCN(C(=O)CCCOC(C)(C)C)C c1(C(N2CCC(C)(NC(C(CC)C(C)C)=O)C2)=O)cc(Br)c(OC)cc1N c1(C(=O)NC(C2CCN(C(c3ccnn3C3CCC3)=O)C2)C)cc(=O)cc(Cl)[nH]1 N1(C(C(C)(O)C2CC2)=O)CC2=C(C1)CN(C(C1(c3ccc(Cl)c(F)c3)CC1)=O)C2 C(=O)(C(O)C(C)(C)C)NCC(CC(C)C)NC(=O)CC1C(C)(C)C1(C)C C(=O)(CC(C)CC(C)C)N1CC(CCC)C(C(=O)NCC2(C)CC3C=CC2C3)C1 CC1CCC(OCCNC(=O)CC2C=CC(NC(=O)Cc3ccoc3)C2)CC1 N1(C(C=CCCCCC)=O)CCCN(Cc2ccc(Br)c(Cl)c2)CC1C Cc1c[nH]c(C(N)=O)c1C(=O)N(O)Cc1cn(C2CC2)nn1 c1(C(=O)OCCC2CC2)c(F)ccc(S(=O)(=O)CC2CC2)c1F C1(C(=O)NCC2(NC(=O)CCn3cc(C)cn3)CCCCC2)(OC)CS(=O)(=O)C1 c1(CCNCCC)c(C)csc1Cl.C(=O)C(F)OC(F)(F)F c1(Cn2cc(CNC(=O)CNC(c3cccc(=O)o3)=O)nn2)ccc(F)cc1 CON(CCC(=O)NCC1CCOCC1C)C(=O)CC(C)(F)F CCCCC(O)C(=O)N1CC2CC1C2C(=O)Nc1cncc(Cl)c1 N1(C(Cc2cc(C)ns2)=O)CC(NC(c2cccc3ccnn23)=O)CC(C)(C)C1 N1(C(c2cc(C)c(F)cc2)=O)CCC2(NC(c3cscn3)=O)CCCC12 C1(C(=O)NCC(C2CCCC2)C)CN(C(=O)Cn2c(O)nnc2O)CCN1C C1(C(N2CC(C)(C(=O)NCC(C(C)C)C)C2)=O)CCOC(=O)CC1 C1(NC(COC)=O)CN(C(=O)C=C2CC2)CC1OC c1(CC(=O)N(C)CC2COCCN2C(=O)COC2COC2)csc2ccccc12 c1(C(=O)NCC(CC(F)(F)F)NC(COCC)=O)nn(C)c2ccccc2c1=O C=CC1(CC(=O)N(C2CN(C(=O)Cc3cnccn3)CC2F)C)CCOCC1 C1(O)(CC(=O)OCC)CCCN(c2ncc(Br)c(C)n2)C1 c1(C(N(C2CCOC2)CCNC(COCC(C)C)=O)=O)ccncc1F CCCC(C)(C)C(=O)N1C2CCC(C2)C1CC(=O)N(CC(C)OC)C CC1OC2CCC1(NC(C1CC(NC(c3cccs3)=O)C1)=O)C2 CCCCC(CCCC)NC(C1CC2(CC2)C12CCC2)=O CCC(C)(O)C(=O)N1CCCC(CCNC(c2cn(C)c(C)n2)=O)C1 CC1CCC=C1C(=O)NCC1CCCCN1C(c1cnc(C(C)(C)C)o1)=O c1(CC(=O)NC2C(NC(C3(C)CCC3)=O)C2)csc2nc(-c3cccs3)cn12 C(=O)(C1c2ccccc2-c2ccccc21)N1C(C)(CNc2ccnc(F)c2)CC1 Cc1cc(N)c(F)c(C(=O)N(C)CCN(C)C(c2ncsc2C2CC2)=O)c1F N1(C(COCC(=O)NC)=O)CC(C(N)=O)(CNC(C2CC2(C)C(C)C)=O)C1 c1(C(=O)NCC2C(C)(C)C2C(=O)NC2CC2(C)C)ncnc(O)c1F C1(C2CCN(C(C3(Cl)CC3(F)F)=O)CC2)(NC(C2=C(C)S(=O)(=O)CC2)=O)CC1 c1(NC(C2C3(CCN(C(c4cc(SC)oc4)=O)C3)C2)=O)ccc2c(c1)CCC2=O CCC(C)C(O)C(C)C(=O)NC12CC1CN(C(=O)CS(=O)(=O)NC)C2 C1(CNC(CNS(CC)(=O)=O)=O)(CO)CCN(C(c2ccc(SC)cc2)=O)CC1 n1(CC(=O)NCC2CCC(NC(=O)CC3CCOC3)C2)ccc(Br)cc1=O N1(C(=O)OC(C)(C)C)CC(C2CC2)C(F)(c2nc(Cn3cccn3)no2)C1 Cc1ccc2cc(C(=O)N(C(CNC(=O)CN=S(C)(C)=O)C3CC3)C)cn2c1 C1(C(N(C2CCN(C(c3ccnn3C)=O)C2)CC)=O)CC2CSCC(C1)C2 c1(C(N2C(CNC(C3CN(C)C(=O)C3)=O)CC2)=O)cc(F)ccc1-n1ccnc1 C#CCCCCC(C(=O)NC1CCOC1)N1CCn2ncc(CO)c2C1 N1(C(C(CCSC)O)=O)C(CNC(=O)CC2CC3CCC2O3)CC2CCCCC12 c1(CNC(C(C)(C)NC(C2C(C)C2C)=O)=O)cncc(F)c1 Cc1cc(Cl)ccc1C(=O)NC1CC(C)(NC(C2CC23CC(O)C3)=O)C1 C1(C(N2C(CCCC)CCC2)=O)CN(C)CCN1C(c1ccsc1C)=O N1(Cc2c(C)nc[nH]2)CCCC(N(C(=O)Cc2ccccc2F)C)CC1 n1(CC(=O)NC2CC(C)N(C(=O)C=C3CCN(C)C3)C2)cnc2sccc2c1=O c1(C(=O)O)cc(Cl)c(CNC2CCC(C(=O)NCc3cccc(F)c3)C2)c(Cl)c1 CON(C)CCCNC(C1(CNC(c2nnsc2C)=O)CC2(CC2)C1)=O C1(C2CCN(C(C3(C)CC3(F)F)=O)C2)CCCCN1C(=O)CN1CCCCCC1 C1(CNC(c2ccn(CC)n2)=O)COCCN(C(=O)CC2CCC(=O)O2)C1 c1(OC)ccc(C(=O)NC2(C)CCN(C(C3(S(N)(=O)=O)CC3)=O)C2)c(OC)c1 CCCC(C(=O)N(CC)CC1CCCC1)NC(c1cn(C)nn1)=O c1(C(N2C(C)CC(NC(c3cc(C(C)=O)oc3C)=O)C2)=O)cnc2occc2c1 c1(OC)ccc(CC(=O)NCCCCCN(C(=O)CSCC(C)C)C)c(OC)c1 Cc1ccc(C(=O)N(C)CCN2CCN(C(C3CC3(Cl)Cl)=O)CC2)c2c1CCC2 c1(CC)nccn1C(C)CC(=O)NC(CNC(=O)CN1CCCCC1)CCOC c1(OC)nccc2cc(NC(=O)Nc3nnc4n(c3=O)CCCC4)ccc12 N1(C(C(C=C)c2ccccc2)=O)C2CCC1C1CC1(NC(=O)CCSCCC)C2 n1(CC)nnc(C(=O)NC(C2CCN(C(=O)CC3CC4CC4C3)C2)(C)C)c1C C1(NC(C2(N(CC=C)CC=C)CC2)=O)CN(C(=O)CSCCCC)CCC1F C1(C(N(C)CC2C(C)OCC2)=O)CN(C)CCN1C(C1CN2CCC1CC2)=O N1(C(c2c(C)noc2)=O)CCCC(O)(CNC(C2CC2C2CC2)=O)CC1 C(CCCCCS(=O)(=O)CCO)NC(CNC1C(C)N2CCC1CC2)=O C(=O)(C1=COCCC1)NCCn1ccc(C(N2CC(C(CC)CC)C2)=O)c1 c1(OC)ccc(C(CNC(C2CC=CCC2)=O)NC(=O)Cc2cnoc2)cc1 N1(C(C2(CC)CCOC2)=O)CCCN(C(=O)CCn2cc(Cl)cn2)C(C)C1 c1(C(N2CCN(CC)CC2)C(=O)NCCOCC)cn(C)nc1Br CCC(C(=O)NCCC(C)(C)NC(c1cccc(Cc2ccccc2)n1)=O)C(C)O Cc1cc(C(N2CCN(C(c3cc4[nH]ccc4s3)=O)C(C)C2)=O)c(C)cn1 C(C(C)(C(=O)N(C)CC1(CO)CC1)NC(=O)CC1CCOC1(C)C)SC c1(OCC)cccc(NC(=O)CON2CCC(NC(C3CS(=O)(=O)C3)=O)C2)c1 C(=O)(CCCN1CCCCC1)NCCN(CCOC)C(c1coc(Br)n1)=O C12(CNC(CC#N)=O)CCC(NC(c3cc(CCO)on3)=O)(CC1)CO2 N#Cc1ccc(N)c(C(=O)NC2CCCC(NC(c3cccc(F)c3)=O)C2)c1 c1(C(N2CCC(OCCNC(C(C)=C3CC3)=O)CC2)=O)ccc2c(c1)CCN2 c1(C(=O)NC(C)CCCNC(=O)CCc2ccccc2Br)n[nH]c2c1COC2 CN1C(=O)c2ccccc2C1CC(=O)NC1C2CC1CN(C(=O)CS(C)(=O)=O)C2 C(=O)(C1=CC2CCCCCCC12)N(CC(=O)NCC1CCOC1)C1CC1 N1(C(CCC(C)C)=O)CCCC(NC(C2CCN(c3ncccn3)C2)=O)CC1 C1(C(=O)NC2CCN(C(c3onc(C)c3C)=O)CC2O)CC(C)(C)OC(C)(C)C1 CC(C)C1=NOC(C(N2CCN(C(C3CC(O)C3)=O)C(c3ccccn3)C2)=O)C1 c1(C(N(C2CCC(NC(=O)CCC(=O)C3CC3)C2)C)=O)cc(Cl)c(F)cc1F C(N=c1ccc([N+](=O)[O-])c(O)[nH]1)C1C(C)CCN(C(=O)CCS(N)(=O)=O)C1 N1(C(c2cccc(O)n2)=O)CCOCC2(COCCN2C(=O)CCCCCF)C1 C1(CC=C)(C(=O)NCc2cn(CC)nn2)CCCN1C(=O)Cc1cc(C)nn1C C1(C(=O)NOCC2CCOC2)N(C(c2cc3n(n2)CCC3)=O)CC12CCCC2 c1(CC(CNC(=O)CCc2cnoc2)NC(C2(C(N)=O)CCC2)=O)ccccc1 C(C(C)(C)CNC(=O)C(c1cncnc1)C)NC(C(=O)NCCOCCOC)=O C1(CNC(Cn2ncc(C)c2)=O)CCCCN1C(=O)C(C1CCC(=O)N1)C Cc1nn(C)c(C)c1C(C)C(=O)N(CCN(c1nccnc1F)C)C(C)C c1(NC(C2COCCN(C(C3(Br)CCC3)=O)C2)=O)ccc(Cl)c(C(F)(F)F)c1 C1(NC(CSCCC)=O)CN(C(c2scnc2C(F)F)=O)CC1OC C1(NC(C(C)C2CCC2)=O)CCC12CCN(C(=O)CCc1ccc(O)nn1)CC2 N#Cc1ccccc1OCC(=O)NC1CC1NC(C1CCN(C2CC2)S1(=O)=O)=O CON1CCC(C(=O)NCCOC2CCN(C(c3cnc(C)c(N)c3)=O)C2)CC1 c1(C(=O)NC(C2CC(NC(=O)Cn3ncnn3)C(O)C2)C)coc2c1COC2 N1(C(C)=O)CCCC(C(N2CC(CCCCNC(=O)C(C)(C)CF)C2)=O)C1 CC1(C)C=C(C(=O)NCC2COCC2NC(c2cc(-c3cccnc3)no2)=O)C1 C(=O)(C(C)(O)C(F)(F)F)N(CCC(C)NC(c1c(C(C)C)nns1)=O)C CC1CCCN(C(=O)CN(C)C2CC2)C1CCNC(=O)Cc1ccnc(OC)c1 C#CC1CN(C(=O)C(O)C(C)C)CCN1C(=O)CCc1ccccn1 C12(CNC(C3C(NC(=O)COC4CCOCC4)CCOC3)=O)CCC(F)(CC1)C2 Cc1ccccc1C=CC(=O)NCCCNC(=O)Cc1cnccn1 CC(C)(C)C#CCCNC(C1CC1CNC(=O)COc1ccccc1)=O C(C1CCCCC1)=CC(=O)NC1CCN(C(=O)Cc2cc[nH]n2)C1C1CC1 C1(c2cn(C3C=CCN(Cc4nc(SCC)oc4)C3)nn2)CCC(C)=CC1C c1(C(=O)NC2CN(C(C(CC)C)=O)CC2C#N)cc(OC)c(O)c(C(C)(C)C)c1 C(=O)(CC(F)(F)CC(=O)N1CCCC1C1CCN(C(c2ccc(F)o2)=O)C1)OC c1(C(=O)NCCOCCNC(c2cc(C)no2)=O)cc(N)ccc1Cl N1(C(C2C=CCC2)=O)CCC2OCCN(C(c3cc(C(F)(F)F)cc(F)c3)=O)C2C1 C1(N(C(Cn2ccc(C)n2)=O)C)CN(C(=O)CCN2CCC(O)CC2)CC12CC2 N1(C(c2c(CC)nco2)=O)CCC(NC(c2cc(N)nc(Cl)c2)=O)C(C(C)C)C1 Cc1cccc(C2(C(=O)NC(C3CCN(C(c4c(Br)cnn4C)=O)C3)C)CC2)c1 Cc1cccc(N(CCC#N)C(=O)NCc2sc(Br)nc2C)c1C C1(NC(C2ON=C(C)C2)=O)CC2(CCCN(C(=O)Cn3cncn3)C2)C1 Cc1ncc(C(C(=O)NCCCC2CC2)N(C2CC2)Cc2nncn2C)[nH]1 C1(N(CC(=O)OCCCN(S(C)(=O)=O)C)C)CCC1F C(=O)(C1=NOC(C2(O)COC2)C1)NCC1(F)CC(NC(C2C(C)C2)=O)C1 C(=O)(C(CNC(=O)C(C)Cn1cccn1)C(C)(C)C)N(CCCC)CCCC C1(C(N2CCC(OCC(C)C)C2)=O)CCCCN(C(c2ncc(F)cc2F)=O)C1 C(C)(C)(C(=O)NCCN(C(C1CC(C)C1)=O)CC1CC1)OCCC N1(C(c2c(OCC)ccs2)=O)CCCC(CCNC(=O)C(C)C(C)C)C1 C1(SCCN(C(=O)C(Cl)Cl)Cc2nc(-c3ccc(F)s3)no2)CCS(=O)(=O)C1 Cc1c(C(=O)NC(CO)C(=O)NCc2noc(C(N)=O)n2)cccc1O C1(C(N2CC(C(C)NC(C(CC=C)CC)=O)C2)=O)CN(C)CCN(C)C1 C(=O)(C(C(C)C)NC(N)=O)NCC1(O)CC(CNC(c2cc(CC)on2)=O)C1 C=C(C)CC(C)C(=O)N1CC(C2(NC(=O)C(CC)OC)CC2)C1 C(C(CC(F)(F)F)NC(=O)CCC1CC1)NC(CCc1nnc(C)n1C)=O c1(CNC(C(CC)(F)F)c2ccco2)cc(-c2nn[nH]n2)cc(S(C)(=O)=O)c1 N1(C(c2coc(OC)n2)=O)CCC(N(c2ccccc2)C)CC1C C12(CCNC(=O)C=CBr)CCC1CN(C(C1CC(F)(F)CS1)=O)C2 c1(C(N2CCC3(NC(C(C4CCCCC4)C)=O)C(C2)C3)=O)c(O)cc(F)cc1F C(C)(C(C)C(=O)NC(C)Cc1cn[nH]c1)NC(C1(CCOC)CCC1)=O C(=O)(C(=O)N=S(C)(C)=O)NCC(CNC(c1c(OC)ccnc1)=O)OC Cc1nc(C(=O)NCC(C2CC2)NC(=O)C(C)n2cncn2)c2ccccn12 Cc1cc(C(N2CC(O)(CNC(=O)C(CO)c3ccccc3)C2)=O)nn1CCO N1(C(CCc2cn(C)nn2)=O)CCC(C(F)CNC(=O)COC2CCC2)CC1 CC(C)(CCNC(=O)CCCCC1CC1)C(=O)N1CCC(CN=[N+]=[N-])CC1 c1(N2CCC(N(C(=O)CCn3cccn3)CCC)C2)nc2ccccc2s1 C1(NC(C(C)SCCCC)=O)(CNC(C2(C(C)C)COC2)=O)CCOCC1 C1(C(=O)NC(CCCCNC(CCC2C(C)=NOC2=O)=O)C)COC2COCC12 C(CCOc1ccccc1)(C(=O)O)NC(CN(C1CCC1)C(C)=O)=O.OCC C1(OC)CCCC1NC(c1cn(C2CCN(C(=O)CN3CC4CC4C3)C2)nn1)=O C#CC1CN(C(C2CC(CC)C2)=O)CCN1C(c1cncc(CO)c1)=O c1(NC(C2C(O)CCN2C(c2c(Br)cccc2Br)=O)=O)nc(Br)ccc1Br c1(NC(c2n(CC)nnn2)(C)CC2CCCC2)cnc2n1CC(C(F)(F)F)CC2 c1(CNC(C=CC(CC)C)=O)cn(C2CCN(C(C3COC3)=O)C2)nn1 N1(C(c2cccc(C)c2Cl)=O)CC2CCOC2(CNC(c2c(C)noc2N)=O)C1 C(C(O)C=CC(=O)NCCCN(C(=O)C(F)C1CCC1)CCO)NS(N)(=O)=O C1(CCOC)(NC(=O)CSc2ccccc2)CN(C(c2oncc2COC)=O)C1 Cc1c(O)cc(C(=O)NC2CCC(C(=O)NCCN(C)CCN)CC2)cc1O CC(C)CC(CNC(=O)CC=C(Cl)Cl)C(=O)NCC1(n2cccn2)CC1 C1(C(N(CCC(C(C)C)N(C)C)C)=O)CCC(C2CCC2)CC1.C12(CC1)C(=O)N2 N1(c2n(C3CC=CC3)nnn2)CCc2cccc(Cl)c2C1 N1(C(CCCNC(C)=O)=O)CCC(CN(C(=O)CC2CCOC2C)C2CC2)CC1 CC(=O)CCCCC(=O)NC1(C(=O)NC2CCN(C)CC2)CCSC1 Cc1cccc(CNC(C2CC3CC3N2C(=O)C=CC2CCOC2)=O)c1O C(=O)(CCCC1CCC1)NCC(C)CNC(=O)COCC1CCCO1 c1(NC2(C)CCN(C(=O)NC(C)C(C)S(C)(=O)=O)C2)ccc(C#N)c(Cl)c1 C1(C(=O)NCc2cccc(C)c2)CN(C(c2cc(C)no2)=O)CC1(C)C Cc1c(C(=O)N(CCC(C)NC(=O)C(O)C2CC2)C)sc(Cl)c1Cl S(=O)(=O)(c1cc(C(=O)NCC(O)CNC(C2(OC)CCC2)=O)c(C)o1)NC C=CCC(CC)C(=O)NC(C1(C(=O)NC(C)C(C)(C)CO)CC1)C c1(C(N2CCC(C3N(C(Cn4c(C)ncc4)=O)CCCC3)C2)=O)ncc(F)cc1N C1(C(=O)NCC2CCCN(C(c3nc(C)oc3)=O)C2)CCC2C(C1)C2(F)F Cc1ccc2ncn(CC(=O)NCC3CCC(C)N(C(=O)C4=CCOC4)C3)c2c1 c1(CCC(=O)NCCSCCN2CCC2)csc(Br)c1.C1(=O)CO1 c1(NC(C(=O)NC(C#C)COC)=O)cc(C)nn1CC1CCCO1 c1(-c2nc(Cc3c(OC)ccnc3)nn2CCCCO)cnc2[nH]ccc2n1 c12ccc(c([N+](=O)[O-])c1)c(=O)[nH]2.c1(C(C)O)n[nH]c(Cn2cccn2)n1 C1(COC)(NC(c2nc(C3CC3)cs2)=O)CCN(C(c2cnsn2)=O)CC1 C(=O)(C(C#N)C(C)C)NC(CCN(C(CCOC(C)C)=O)C)C(C)C C1(NC(C=CC2CCN(C(CC3(C=C)CCC3)=O)CC2)=O)CCn2cncc2C1 N1(S(c2ccc(OCC)cc2)(=O)=O)Cc2cc(Br)ccc2CC1C c1(NC(C2CCCN(c3nc(=N)[nH]cc3)C2)=O)c(N2CCCCC2)ncnc1Cl c1(CNC(N(C)Cc2nccn2C2CC2)=O)cc(C(F)(F)F)ccn1 C1(CN(C(C(C)=CC)=O)CC)CCCN1C(=O)C(CC)NC(N)=O C1(CNC(CCN(C(C(COC)COC)=O)C)=O)OC(=O)CC1(C)C C1(NC(=O)COC2COC2)CCC(NC(C2CCCO2)=O)CC1 c1(C(C)(C)C)ncc(Br)c(N2CC3C(NC(c4cc(Br)cs4)=O)C3C2)n1 Cc1n[nH]c(C)c1CC(C)C(=O)NC1CCN(C(c2cnc(Cl)n2C)=O)C1 C1(NC(c2cccc(CNC(C)=O)c2)=O)CC2CC1N(C(c1ccncn1)=O)C2 N1(C(CC(C)C)=O)CC2CC(CNC(c3cc(C(N)=O)ccc3Cl)=O)C2C1 N1(CC(C)C)CC(C(=O)Nc2cccc(Cn3cc(C4CC4)nn3)c2)CC1=O C1(C(C)OC)CCN(C(C23CC2CCN3C(C2CC(C)CCO2)=O)=O)CC1 C=CC1OCCCC1C(=O)NC1CC(NC(C2Cc3cscc3C2)=O)C1 C=C(C)C1CN(C(=O)C(C)C(C)NC(c2cc(C3CC3)on2)=O)CCO1 C1(C(=O)NCCN(C(CC)C)C)CC2CC1CC2NC(=O)C#CC(C)(C)C CCC(C(=O)OC)C(=O)N1CCC(n2cc(-c3cc(F)ccc3C)nn2)CC1 c1(OC)nn(C)cc1CNC(=O)CC1CC(C)N(C(=O)CC(Cl)Cl)C1 C(C(O)CC(C)(C)C)NC(CC1(N(C(=O)Cc2ccnn2C)C)CC1)=O C(=O)(C#CC1CC(F)(F)C1)N1CCN(C(C=CC=CCCCCC)=O)C(C)C1 c1(CC(N2CCC(C(N3CCC(O)(CO)C3)=O)C2)=O)ccc(F)c(Cl)c1 C1(NC(C(CSC)OC)=O)CS(=O)(=O)CC1NC(c1cn(CCO)nn1)=O C1(CCC(=O)NC2CC(NC(COCCN(C)C)=O)C2)CCN(C)CC1 Cc1cccc(CCC(=O)N2CC(n3cc(-c4cnn(CCF)c4)nn3)C2)c1 CCC(CNC(=O)CCCC#N)(CC)NC(=O)C(=O)NCC1CC1 C1(C)(NC(C2CCC(N(C)C)CC2)=O)CCCN(C(=O)CC2CC2(Cl)Cl)C1 Nc1cccc(F)c1C(=O)NCC1CCCCN1C(=O)Cc1cncnc1O C1(C(=O)NCCN(C(C)=O)C)CCC(C(N)=O)CC1.C12(CC1)C(=O)O2 N1(CCCNC(C(COC)OC)=O)CCN(C(C23CCC(CC2)O3)=O)CC1 C(=O)(N=c1[nH][nH]cc1C(F)(F)F)C12C(CN(C(=O)Cc3cc(Br)ccc3O)C1)C2 O=C(CN=c1cc[nH]cc1)NC1CCN(C(=O)CCCCF)CCC1CO c1(OC)ccc(C(N2CC(CNC(c3cncs3)=O)C3CC23)=O)c(F)c1 C1(C(N2CCN(c3ccccc3)CC2)=O)CN(Cc2cscc2OCCO)CCS1 C12(NC(C3=NNC(=O)C3)=O)CCCC1N(C(C13CCC(C(F)F)(CC1)C3)=O)CC2 n1(CC(=O)NC23CC2CN(C(=O)CCCn2ccnc2)C3)ncc2cccnc12 c1(SC)nc(C)cc(=NCC2CCC3(CCC3)C2NC(=O)CC(C)C)[nH]1 C1(CC(N2CCOCC(NC(C3(CO)CCCC3)=O)C2)=O)CCC2(CCC2)OC1 C1(O)(CNC(=O)COCC2CCC2)CCCN(C(c2ccc(Cl)o2)=O)CC1 C(=O)(C=C1SCC(=O)N1C)NC1CN(C(C(C)OCCC(C)C)=O)CC12CCC2 C=CCC(COC)N=c1[nH]c(=NCC2(C)NC(=O)NC2=O)c2ccccc2[nH]1 C#CC(C)(C)C(=O)N1CCOC(C(=O)NCC2(C#N)CC2)C1 CC1CN(C(=O)CC(c2ccc(Cl)cc2)O)CCN1C(c1cc(C2CC2)ns1)=O Cc1c([N+](=O)[O-])c(CC(=O)NCC2CCCCCN2C(=O)OC(C)(C)C)nn1C c1(OC)ccsc1C(=O)NCCC1CCN(C(=O)CCSCC(N)=O)C1 C(=O)(C(O)C(C)C)N(CCNC(C(CO)OC)=O)C C12(NC(C(C3CN(C(C45CCC(CC4F)C5)=O)C3)OC)=O)CC1COC2(C)C C(=O)(C(C#N)C(C)(C)C)N1C(CC(=O)NCC2CCC(C)(C)CC2)CCC1 C=CC(C(=O)N(CC(C)NC(=O)Cn1ccc(CC2CC2)n1)COC(C)(C)C)OC c1(CC)cc(C(N2CC(CNC(C3CN(C(C)C)C3)=O)C3CC23)=O)c(C)o1 c1(CC(=O)NCCC(C)N(C)C(c2ncn(C)n2)=O)ccnc(F)c1 C1(C(N(C23CC(C2)C3)CC)=O)COC2(C1)CN(C(c1cccc(C#N)c1)=O)C2 Cc1nn[nH]c1C(=O)N(CCNC(=O)CCC#N)Cc1ccccc1 C(CCC(=O)NCCCOCCC(N1CCCC1CN(C)C)=O)=C(C)C N1(C(c2cc(C)c(Cl)cc2F)=O)CCN(C(=O)Cc2ccco2)C2CCCCC12 c1(C(C(=O)NCCN(CC(C)O)C(C2C(C#C)C2)=O)(F)F)ccc(C)cc1 N1(c2ncc(C#N)cc2Cl)CCC2(CC1)COC(CNC(C1(Cl)CC1)=O)C2 C1(C)(CNC(CN(CC)CC)=O)CN(C(c2oc(C(C)=O)cc2C)=O)CCO1 C1(OCC(=O)NC(C)CC2CN(C(=O)CSc3nncs3)C2)CCC(F)(F)CC1 N1(CC(=O)NC(c2ccc(OC)c(F)c2)C(F)(F)F)c2ccccc2NS1(=O)=O Cc1ccnc2c(NC(C3NC(=O)OC3C)=O)cccc12 C(=O)(C1=NOC(C)C1C)NC1CCCC(NC(Cn2c(C)nc(C)n2)=O)C1 c1(NC(C2CC(NCc3cc(Br)cc(I)c3)C2)=O)ccc(I)c(Br)c1 c1(C(=O)NCC2(OC)CN(C(c3ccn(CCC)n3)=O)C2)cc(=O)c(OC)c[nH]1 Cc1cscc1Cn1cc(CC(C(=O)O)NC(=O)C(c2ccccc2)F)nn1 CCC(CCC(=O)N1CCCC1)NC(C1CN2CCN1CC2)=O.C1CC(=O)N1 c1(CC)c(C(=O)NCC(C)N(C)C(C2CC3(CCC3O)C2)=O)sc2ccccc12 c1(CNC(C=CCC)=O)ccc(CNC(C2(C)CCCCO2)=O)c(F)c1 c1(CC(=O)NCC(CC)NC(C2(C(=O)N(C)C)CC2)=O)csc(-c2nc[nH]n2)n1 C1(C(=O)NCCCC(=O)NC(C)(C)CC2CCOC2)CC(O)C(F)C1 n1(CC(=O)NCC2CCN(C(C(C)c3ccco3)=O)CC2)nnc2ccccc12 c1(C(N2CC(C)(COC)C2)=O)ccc(NC(c2cccnc2)=O)cc1Cl N1(CCCCCSC)CC(N=c2[nH]c(=NC)[nH]c(=NCC3CCC3)[nH]2)CC1=O CC1CCC(C(N2CC(O)(CNC(=O)Cc3ccc(Cl)cc3F)C2)=O)C(=O)N1 c1(CC(C)C)ncc(C(C(=O)NCC2CCOC2)N(C2CCC2)C)s1 N1(C(Cc2cn(C)nc2)=O)CCN(C(c2cnccn2)=O)C(c2ccccc2)C1 N1(C(C(C)C2CC2)=O)CC(C(N2CCCC(NC(=O)C3CC3)C2)=O)OC(C)C1 Cc1ccc(NC(c2occc2C)=O)c(SCn2cncn2)c1.C12CCCN1C2 C1(C)(NC(C2(NC(CCc3cn(C)nc3)=O)CSC2)=O)CS(=O)(=O)C1 C1(NC(CNC(C(CC)C)=O)=O)CCN(C(=O)CC2CCCC2O)C12CC2 N1(CCNC(=O)C(Cc2ccoc2)NC(C23CC(CO)(C2)C3)=O)CCC(O)CC1 C1(C(=O)NC2CN(C(c3c(OCC=C)cc(Cl)cc3)=O)C2)CC1C1CCOCC1 C(=O)(C(C)(C)C(=O)NCCCN(C)C(C1CN(Cc2ccccc2)C1)=O)OC N1(C(c2c(CC)csc2)=O)CCC(C(F)F)(CNC(C2CC2C(F)(F)F)=O)C1 N1(C(c2c(CC)ocn2)=O)CC2CC1CN(C(C1CCS(=O)(=O)C1(C)C)=O)C2 c1(CN2C(C(=O)Nc3cnc4sccc4c3)COCC2)c(F)cccc1[N+](=O)[O-] NS(=O)(=O)c1coc(C(N2CC3CCC3(NC(C3CC3F)=O)C2)=O)c1 CCCC(CC)C(=O)NCCCC1CN(C(C23CC4CC2C3C4)=O)CCO1 C1(CNC(COCc2cc(C)no2)=O)CC2CCC1N2C(c1csnc1Cl)=O C12CN(CCO1)C(=O)CNC2.c1(C(C)=O)cnc(CC(C)(C)C)o1 CCC(C)CN=c1nc(N2CCN(CC(=O)N(C)C)CC2)c2c([nH]1)CCC(C)C2 C(C(CC(C)C)NC(C1CC1c1cn[nH]c1)=O)NC(c1cc(C)ns1)=O C(=O)(C#CC1(CC)COC1)NC1(CC=C)CCN(C(c2ccc(O)nc2Cl)=O)C1 c1(C(N(CC(C)O)CCNC(C2CC2F)=O)=O)cc(C(N)=O)cc([N+](=O)[O-])c1 c1(C(=O)NC2(C#C)CCCC2)ccc2c(c1)N(C(=O)OC(C)(C)C)CCS2 C1(NC(C2N(CCC)CCCC2)=O)CC2(CCCCN2C(C2CCC2)=O)C1 C1(CC(=O)OC)(CCNC2CCN(C(N3CCCC3)=O)C2)CCCC1 N1(C(c2cccs2)=O)CCC(C2CCCN2C(c2csc(Cl)n2)=O)C1 Cc1cc(C(=O)NCC(C)(C)CNC(c2nccc(Cl)c2C)=O)nc(C)c1 c1(CC)ccc(C(=O)NC2CCC(C)(NC(=O)CCCC3CCC3)CC2)cc1F C1(CC(=O)NC2CN(C(C3CCCC(OC)C3)=O)CC2C)CC2CCC(C1)N2C CC(CC(F)F)C(=O)NC12CC(CNC(=O)CCC3CCCO3)(C1)C2 c1(OC)cc(C)c(-c2ccc(C3CN(C(C4CC5(CCC5)C4)=O)CCO3)cc2)cn1 CC1CN2CCN1C(C(=O)NC1CC(NC(c3ccc(F)c(O)c3F)=O)C1)C2 N1(C(CC=CC=C)=O)CCCC(N(C)C(c2cc(C(N)=O)ccc2OC)=O)CC1 CC1(C)Cc2ccccc2CN1CC(=O)NC1CC(F)(F)C12CC2 C(=O)(C1=NN(C)C(=O)CC1)N1CCN(C(C(CC)O)=O)C(C2CC2)C1 c1(C(N(C2CCN(C(C3CNC(=O)C3)=O)C2)CC)=O)csc(C(F)F)c1 CCCC(CNC(=O)CCc1cncs1)NC(C12CC(C1)C2)=O C=CC1(C(=O)NCCn2cc(C)cn2)CCN(C(=O)C(O)C2CCCC2)CC1 c1(C(=O)NC(CN(C(C2(NC(C)=O)CCCCC2)=O)CC)C)nc(Cl)ccc1N c1(-n2cc(CN3CCCC(NC(C=CS(C)=O)=O)C3)nn2)ccc(F)c(Cl)c1 c1(C(N(C2CN(C(=O)CCc3nc[nH]n3)CC2F)C)=O)cncc(F)c1 CCCC(C(=O)NCCCN(c1ccnc(-c2ccccc2)n1)C(C)C)OCC C1(NC(CCC(=O)NC)=O)CC2CC(NC(c3cnccc3C)=O)CC12 CCCCC(O)C(C)C(=O)NC(CCC(=O)NC(C)(CC1CC1)C1CC1)C(C)C C1(C(N(CCS(C)(=O)=O)C)=O)CCN(C(C2(CCF)CCC2)=O)CCO1 N1(C(C2C(CNC(COc3cn(C)nc3)=O)CCCC2)=O)CCc2c[nH]nc2C1 C1(NC(=O)CC2C=CC(NC(=O)C(O)Cn3cncn3)C2)CNC(=O)OC1 N1(C(CC(C)C)=O)Cc2ccnn2CC(NC(=O)C(F)C(C)(C)O)C1 C1(NC(c2cc(C)c(Cl)s2)=O)CN(C(c2ncoc2C(C)C)=O)CC1C1CC1 C(=O)(CC(C)F)N1CC(C(C(=O)NCCNS(N)(=O)=O)OC)C1 N1(C(c2c(C)con2)=O)CC(C)(C(N2CC3(CCC2CO)CC3)=O)CC1(C)C c1(C(=O)NC2(C)C(C)C2)ccc(CNC(C2OCCC2(C)C)=O)nc1 C(=O)(C1=NOC(C)(C)C1)NCC1N(C(c2cc(C)c(Br)s2)=O)CC2(CC2)C1 N1(C(CCCC)=O)CCN(C(c2nc(C)nn2C)=O)C(c2cccnc2)C1 N1(C(c2ccc(OC)cc2C(F)(F)F)=O)CC(C(=O)O)CC(C)(C)C1 c1(C(=O)NC(CNC(C2C(COC)C2)=O)CO)cc(Cl)c(Cl)c(Cl)c1 c1(C(=O)NCC2C(NC(c3n(C)nnc3)=O)C2)csc(Cl)c1Cl c1(C(=O)NC(C)C2=NOC3COCC23)cnc2c(cnn2C)c1N N1(C(c2cc(C(C)=O)c(C)o2)=O)CCC(NC(c2n[nH]cc2Cl)=O)C(CO)C1 c1(C(=O)OC)cccc(CNC(C2CCCC(Nc3ccnc(C)n3)C2)=O)c1 S(=O)(=O)(c1cccc(F)c1)NCC(N1C(NC(=O)CC2CC3(COC3)C2)CC1)=O N1(C(CCOCCC)=O)CCCC2(CCN(C(c3cc(C)n(C(F)F)n3)=O)C2)C1 c1(-c2n(CC)nc(CCSC)n2)ccc(N2CCOCC2)c([N+](=O)[O-])c1 N1(C(C2(C)CCCOC2)=O)CC2CCC(NC(c3csc(C4CC4)n3)=O)CC2C1 c1(CCOC)nnc(N(C(C)CNC(=O)CC2CC(F)(F)C2)C)s1 S(=O)(=O)(c1cccnc1NC1CC(=O)N(C2CC2)C1)NCC(CC)O c1(OC)cccc(C(=O)NCC(O)CCNC(C2CC2c2ccn(C)n2)=O)c1C CC(C)C(C)(O)CNC(=O)C(c1cccs1)NC(c1cnnc(O)c1)=O c1(CC)cc(CC(=O)NCC2CC(NC(C3CSCN3C(C)=O)=O)C2)n(C)n1 N1(C(CCC=CC)=O)CCN(C(=O)Cc2c[nH]c3cccnc23)C(C)C1C N1(C(C(C)(C)C2CCCO2)=O)CC2CC2(CNC(c2ccncc2F)=O)C1 CC1(C(=O)NOCC2CCOC2)C=CCN1C(C1CCSCC1)=O C1(NC(C2C(C)C2)=O)CCC2CC1CN2C(=O)C=Cc1ccc(=N)[nH]c1 C1(N(C)C(c2cnco2)=O)CCCC(N(C)C(c2ccnc(O)c2)=O)C1 c1(C(N2CC(F)CC(NC(C=C(C)c3cccs3)=O)C2)=O)ccc2nncn2c1 c1(C(N2C(CNC(=O)CC3CC=CCC3)CCC2)=O)cc2c(=O)cc[nH]c2s1 C(=O)(C1CCCc2scnc21)NC1C(NC(Cc2c(C)ccs2)=O)CC1 C1(CNC(Cn2cc(-c3onc(C)n3)nc2)=O)COCCN1C(=O)C(C)C c1(CC)ncccc1C(=O)N(CC(=O)NC1CCC1)Cc1ccc(F)cc1 n1(CC(=O)NCCCOCCN(C)C(C2CC(CF)C2)=O)ncnn1 Cc1nc(C(N2CCSCC2CCNC(C2CCC(N(C)C)C2)=O)=O)c(C)n1C Cc1cc(C(C(=O)NC2CCOCC2)N(CCSc2ccccc2)C)cnc1C C(=O)(CC(C)C(C)(C)C)N(CC(C)CNC(C1CC(S(C)(=O)=O)C1)=O)C N1(C(c2cc(C)oc2C(F)(F)F)=O)CCN(S(=O)(=O)CC2CCC2)C(CC#N)C1 C#CC(C(C)C)NC(c1conc1C(C)NC(c1cc(CCO)on1)=O)=O c1(C(N(CC(C)NC(CC2CCC(C)CC2)=O)C)=O)cc(Br)ccc1N C12(C(NOCC(N3CC(c4nc[nH]n4)(CC=C(C)C)C3)=O)=O)CC(CCO1)C2 N#CC1CN(Cc2ccc(C(F)(F)F)cn2)CCN1C(c1cccc(O)c1F)=O N1(C(CC=CCC)=O)CC2(C1)OCc1cc(-c3cc(OC)cc(F)c3)ccc12 c1(C(=O)NCC(CNC(CC2CC(OC)C2)=O)(C)O)ccnc2ccnn12 Cc1c(C(=O)NCC2CC2NC(C2CC3(C2)CC(O)C3)=O)[nH]c2c1CCCC2 C1(CNC(C(N)=O)=O)Cc2ccccc2CN1C(=O)C(F)CC1CCC1 N1(C(c2cccc(F)n2)=O)CCC2(C1)CN(C(c1ncoc1C(F)(F)F)=O)C2 Cc1cc(=NCC2CCC3CC2C3(C)C)[nH]c(=NCC(=O)N2CCCO2)[nH]1 C(C(=O)N=c1ccn(CC)[nH]1)N(C(=O)C(CCC)N(C)C)CC#C c1(NC(N2CC3(OCC(C(=O)OCC)C3)C2)=O)cnc(O)c2c1NCCC2 C1(NC(CN2CC(C)C2)=O)CC2CC1N(C(C1(C)CC=CCC1)=O)C2 c1(C(C)(C)C)cccc(C(=O)NC2C=CCN(C(=O)Cn3ccnn3)C2)n1 N1(C(c2ccc(CC(C)C)nc2)=O)CC2(C1)CN(C(=O)C(F)=C1CCC1)C2 C(=O)(C(=O)N=S(C)(C)=O)N1CCC(O)(C(C)NC(c2cc(=O)n(C)cn2)=O)C1 C1(C(=O)NC(C(=O)NCCCc2cnn[nH]2)C2CC2)CC12CCOCC2 C1(C(=O)NCC2N(C(=O)CC(O)CN3CCOCC3)CC2)CC2(COCCO2)C1 Cc1ccnc(C(=O)NC2CCCCC2CNC(c2snnc2C)=O)c1N c1(CN2C(C(N3CCC(C(N)=O)CC3)=O)C3CCC2C3)cc(O)c(Br)cc1O c1(N(C2CC23CCNCC3)C(c2ccc(OC)cc2OC)=O)ccn2nccc2n1 c1(C(=O)NC(C2CCCCC2)C(C)NC(C2CC(F)(CO)C2)=O)ncncc1Cl C(C(C)(C)C(=O)NCC1CC(NC(=O)CCc2ccc[nH]2)C1(C)C)OCC N1(CCCC)C(=S)NC(c2c(N)cnc(Cl)c2Cl)C(C(F)(F)F)C1(O)CCCOC c1(CC)ncc(C(N2CCC(N(C(=O)C(F)(F)COC)CC)CC2)=O)c(O)n1 c1(OC)ccn2cc(C(N3CC(C4CN(C(C5CNC(=O)N5)=O)C4)C3)=O)nc2c1 C1(NC(c2c[nH]c(-c3ccncc3)n2)=O)CC2CN(C(C3CSC3)=O)CC2C1 C1(n2cc(C(C)OC)nn2)CCC(CNC(C2CCOCC2)=O)CC1 C1(C)(CC(=O)NC(CC)CN(C)CC)CCN1C(C1CCCCC1)=O c1(N2CC3(CN(C(CS(CCC)(=O)=O)=O)C3)C2)ccnc2nc(C)nn12 N(C(=NCCC(C)=O)NC1CCN1c1ccc(Cl)cc1)CC(C)OC N(C(=NCC1CC1)NCc1cccc(Br)n1)CCCC=C(C)C Cc1ccc(S(=O)(=O)NCCCNC(c2ccc(-c3cnco3)cc2)=O)cc1 C1(NC(C2=NOC(C)C2)=O)CCC2CN(C(c3ccc(F)c(Cl)c3)=O)CC2C1 c1(C(N2CC3CCN(C(=O)C4=CCS(=O)(=O)C4)CC32)=O)c[nH]c2cc(F)ccc12 c1(CC(=O)N(CCCNC(C2=C(C)CCC2)=O)C2CC2)ccc2c[nH]nc2c1 c1(OC)cc(C2CCCN(C(=O)C(C3CCS(=O)(=O)CC3)NC)C2)ccc1F Cc1cc(C)c(C(=O)NC(C(=O)NOC2CC3CCC2C3)C2(O)CCC2)o1 Cc1nc(C(=O)NC2CC(CC(=O)Nc3[nH]cnc3C#N)C2)ccc1F C1(C(=O)NCCCCCNC(C2(OCC)CCOCC2)=O)CCn2cnnc2C1 c1(C(N2CCC(N(C(=O)C=CCOC)CCC)C2)=O)sc(=NCC)[nH]c1C C1(C)(CC)CCN(Cc2coc(-c3ccccc3)n2)C1 CC1C(C(=O)NCC2(O)CN(C(=O)C(C)(F)F)C2)C1(F)F N1(C(c2nnn(C)n2)=O)CC2C3CCC(C2C1)N(C(c1cncc(N)n1)=O)C3 C1(OC)(CNC(C2CC(=C3CC3)C2)=O)CCN(C(=O)CN2CCCCC2)C1 c1(C(=O)NCC(CNC(CC)=O)(C)OC)ccn2nncc2c1 C(=O)(C1c2c[nH]nc2CN1C(=O)CCCn1cccn1)NCCC(=C)C Cc1nsc(C(=O)NCC2(C)CCCN2Cc2ccccc2)c1Br c1(C(=O)NCCOC2CN(C(C(C)SCCCC)=O)C2)c(F)ccc(F)c1O C1(C)(C(N2CC(CNC(C)=O)C2)=O)CCN(C)C1=O.N12CCN(CC1)CC2=O C(=O)(C(F)C(F)(F)C(F)(F)F)NC(CNC(c1n(CC)c(O)nc1)=O)CCOC C(=O)(CS(=O)(=O)c1nnc(-c2ccccc2)n1CC1CC1)Nc1c(CC)ocn1 N1(C(C2C(C(=O)OC)CC2)=O)CC(F)CC1CNC(=O)CCc1ccccc1C C=CCC(CC)C(=O)NCc1ncoc1CCNC(=O)CC1CCOC1=O C1(C(N2CCC(C)C(CNC(=O)C3=CCCSC3)C2)=O)C(C)(C)CCCC1(C)C c1(-c2c(C)noc2)cnn2c1CN(C(c1cccn3c(O)nnc13)=O)CC2 CC(=O)CCCCC(=O)N1CCC2(CC2)CC1C(=O)NC1CCCC2(CC1)CC2 N1(CCC2CCN(C(=O)OC(C)(C)C)C2)CCC2(CC1)CCS(=N)(=O)C2 N1(C(c2c(CC)non2)=O)CCOC(CNC(=O)CC2C=CCC2)C1 C(CCCN=[N+]=[N-])NC(COC1CCN(C(C(C)CC2CCC2)=O)C1)=O Cc1nc2sccn2c1C(=O)NC1CC1NC(c1cnc2cnccc2c1)=O C1(NC(c2cn(CC)nc2)=O)CC2(C1)CC(NC(=O)C(c1ccc(F)cc1)C)C2 N1(C(CCSCC)=O)C2CCC1CC(N(C)C(C1CCCN(C(=O)CC)C1)=O)C2 c1(C(=O)OC)ccc(C(=O)NCCCN(C(=O)CCC2CCN(C)C2)C)cc1O C1(NC(C2CN3CCC2C3)=O)CCCC(C(=O)NOCC2CC(F)(F)C2)C1 C1(C)(NC(c2cc(C)c(C)o2)=O)CCCN(C(C2CN(C3CCOC3)C2)=O)C1 N#Cc1cccc(CC(N2CCCOC(CCNC(c3ccsn3)=O)C2)=O)c1 c1(C(CCC)NC(=O)C(Cc2cccc(C)c2)CC)cccc(S(=O)(=O)NC)c1 N1(C(COCC=C)=O)CC(F)(F)CC1CCNC(=O)C(C)CC(F)F c1(C(N2C(CNC(CN(C(C)=O)C)=O)C=CC2)=O)nn(C)c(Cl)c1Br N1(C(C(C)SCC)=O)CCN(C(=O)CCC(=O)c2cnn(C)c2)C(CF)C1 n1(CC(N2CC(NC(C(C)OCCC=C)=O)C(F)C2)=O)ccc(=O)c([N+](=O)[O-])c1 C1(NC(=O)CC2CCSCC2)CCCCC1NC(C1(CF)COC1)=O c1(C(=O)NC(CNC(C2CCCN(C)C2)=O)CO)cccc2c1nc(O)n2C Cc1cc(=NC2CC2C(C)C)[nH]c(NC(c2ccc(Cl)cc2)Cn2cnnc2)n1 C1(CC=C)(NC(=O)C(F)C2CCOC2)CCN(C(c2snnc2C)=O)CC1 N1(C(c2c[nH]c(=NC)s2)=O)CC2(CCN(C(c3n[nH]c4c3CC3CC43)=O)CC2)C1 Cc1cc(C(=O)N(C(C)CN(C(=O)Cn2cnc([N+](=O)[O-])c2)C)C)ccc1F N1(c2c(C(=O)OC(C)C)cccn2)C2CCC1CC(NC(=O)C1=COCCO1)C2 C1(C(=O)N(C)Cc2cn(C)cn2)(NC(C2C(C)CC2)=O)CCSC1 C1(C(N2CCC(OCC=C)C2)=O)CN(C(=O)CCc2cncn2C)CC1CCC Cc1ccc2c(c1)C(C(=O)N1CCN(C(=O)C(C)(F)F)CC1)CC2 C=CCC(C(=O)N(C)CCN(C)C(c1ccc(CN=[N+]=[N-])o1)=O)N(C)C C(=O)(C1=NN(CCO)C(=O)CC1)NCC(CNC(c1c(C)cc(F)s1)=O)O C1(CCNC(c2cnc(Cl)cc2Cl)=O)CCCN(C(=O)CCc2cnoc2)CC1 N1(C(C(CCSC)NC(c2ccc(F)cc2)=O)=O)CCc2cc(C#N)ccc2C1 c1(OC)ccc(C(N2CC(CNC(c3cc4c(s3)CCCC4)=O)C2)=O)c(N)c1F c1(C(N2CC(CNC(Cc3cnc(C)o3)=O)C(O)C2)=O)c(C)nc(C)n1O N1(C(CC(C)n2ccnc2)=O)C2CCC1CC(CNC(C1(O)CC1(C)C)=O)C2 c1(C(CO)NC(C2(CO)CC2)=O)ccc(C2CCCCC2)cc1 c1(CCNC(c2cccc(-n3cccc3)c2)=O)c[nH]c(=NCc2cccnc2Cl)s1 N12CC3CC1C3C(=O)NC1CC(C1)C2=O.c1(OC)ccnc(C2CC2)c1 C1(C(=O)NCc2cn[nH]c2)(NC(C(C)c2ccco2)=O)CCC(C)(C)C1 C1(C(=O)NC(CC)CNC(=O)C(c2cccc(Cl)c2)O)CN2CCC1CC2 c1(C(=O)NC23CC(CNC(Cc4nc(C(C)C)sc4)=O)(C2)C3)ccc(O)c(N)n1 C1(NC(COC)=O)CCOCC1NC(=O)C=C1CCSCC1 c1(C(=O)N(C2CCCC(CNc3ncc(Cl)c(O)n3)C2)CC)nccc2nc[nH]c12 C1(NC(CC(n2c(CC)ncc2)C)=O)CC(C)CN(C(=O)CN2CC(C)(C)C2)C1 Cc1cc(C(=O)Nc2cc(Br)nn2C)ccc1OC(c1ccccn1)C Cc1cc(CC(N2CC(O)(CCNC(c3ccc(C)nn3)=O)C2)=O)cc(C)c1 N1(C(=O)C2=CCCSC2)CCCCCC(NC(C2(F)CC=CCC2)=O)C1 C1(CNC(c2n[nH]c(CC)c2Cl)=O)CCC(C)CN1C(c1cscc1Cl)=O C1(NC(c2cccc(F)c2F)=O)CN(C(=O)CC2CCS(=O)(=O)CC2)CC12CC2 C1(CNC(c2n(C(C)C)ncc2)=O)C2CC1N(C(C1CCSC1)=O)C2 Cc1cc(C(N2CC(O)(C(F)C(N3CCC4(CC4)C3)=O)C2)=O)nc(C)c1 c1(OC(c2c(OC)nc(N(C)C)cc2)=O)ccc(S(=O)(=O)N(C)C)cc1 N1(C(c2nn(CCOC)c(=O)cc2)=O)CC2C3CCC(C2C1)N(C(=O)C=C(Cl)Cl)C3 C(=O)(CS(=O)(=O)CC1CCCO1)NC1C(CNC(CN(CC(=O)NC)C2CC2)=O)C1 C1(N(c2ccco2)C=O)CCCC12CN(CC1CC1)C2.c1(-n2ccnn2)cc[nH]c1 C(CC(CNC(c1ccc(CC(C)C)s1)=O)NC(=O)C(c1ccccc1)F)OC C(=O)(C(CCF)NC(C1CCCCN1CC)=O)NCC=C C1(O)(CNC(C2(Cl)C(C)(C)C2)=O)CCCN(C(C2CN(S(N)(=O)=O)C2)=O)CC1 C#Cc1ccc(CC(=O)N(C2CCCC(NC(=O)CS(=O)(=O)N(C)C)C2)C)cc1 Cc1ccnn1CC(=O)NCCNC(c1csc(COc2ccccc2)n1)=O Nc1c(C(N2CCC3(CC(NC(=O)CC4C=CCC4)C3)C2)=O)cc(F)c(F)c1F CCCCC(=O)NC1COCC1CNC(c1ccnn1C(C)C)=O C1(c2cn(C3C(C(=O)OC(C)(C)C)CC(C(=O)O)C3)nn2)CCCCNC1=O N1(C(C2C(C)(C)C2(C)C)=O)CC(NC(c2ccccc2Cl)=O)C(F)(F)C1 Cc1cc(C(=O)NCC2(O)CCN(C(C3COC(=O)N3)=O)CC2)c(C)c(C)c1 C12(NC(CCC)=O)CCCCCC1N(C(=O)C(O)C(C)CC)CC2 C1(C(=O)NCCC(COC)OC)CC2C=CC1N(C(=O)CCCCC(C)C)C2 c1(C(N(CC(CC)NC(=O)C=CCN(CC)CC)C)=O)coc2c1CCCC2 CC(O)CCCCCC(=O)NCC1CCN1C(C1(c2ccccc2)CCOC1)=O CCC(CC(=O)NC1CCC(NC(=O)C(F)(F)Sc2ccc(Cl)cc2)C1)C(F)F c1(SCC(=O)NC(C2CCN(C(=O)CSc3ccncc3)C2)(C)C)ccccn1 C(=O)(CCCCC(=O)N1CC2CC(NC(=O)C=Cc3ccc(C)cc3)C1C2)OC c1(C(=O)NCC2CC(NC(CC(C)(F)F)=O)C(O)C2)cccc2c1NC(=O)CC2 C=CC1CCCCC1.c1(C(=O)NCCOCC=C)cccnc1C(F)F c1(C(N2C3CC(NC(C(CCC)(C)C)=O)C(C3)C2)=O)ccc2cnccc2c1 C1(C(=O)NC(C(C)NC(c2coc(N(C)C)n2)=O)C)CCc2cc(F)ccc2O1 c1(NC(C)=O)sc(Cl)cc1C(=O)NCCC(C)NC(C1CC1(C(C)C)COC)=O N1(C(c2nc(C(=O)OCC)oc2)=O)CC(CNC(=O)CCCNC(C)=O)C(O)C1 C1(C)(C(N2CC(CC)SCC2)=O)CC(O)CN1C(=O)Cn1cc(C2CC2)nn1 S(=O)(=O)(c1cc(Br)ccc1OC)N.c1(C(=O)NCCOCCCC)ccc(Cl)cc1F C(=O)(C1=CCCCCC1)NC1CCCN(C(CCc2cc(C)no2)=O)C1 C1(CNC(=O)C=CC2CCC2)CCN(C(C2CCCN2C2CC2)=O)CC1(F)F C1(NC(c2n(C)nnc2)=O)CCN(C(c2ccc(C3CC3)o2)=O)CC1F Cc1cccc(CC(=O)NCC2CCCCN2C(C2CCCC(C(N)=O)C2)=O)c1 N1(C(C)=O)CCC(C(=O)NCC2CN(C(c3scnc3C)=O)C2)CC1 N1(C(c2nccc(C)n2)=O)CC2CCCCC2(CNC(C2CN(C(N)=O)C2)=O)C1 N1(C(C2C(C=C)C2)=O)CC(NC(=O)CCNS(=O)(=O)CC)CC2(CC2)C1 C1(C)(NC(c2c(CCC)n[nH]c2)=O)CCCCC1C(=O)NCCCC1(O)CCC1 C1(C)(CNC(C(C=CC)O)=O)CCN(C(=O)CCCCNC(=O)OCC)CC1 N1(C(C(C)OCCOC)=O)CCOC(C)(CNC(C2(C)CCC3CC3C2)=O)C1 N(C1CN(C(=O)C2CCc3nccn32)Cc2ccccc21)C(C=COCC)=O CC1(C)CC(CNC(=O)CS(N)(=O)=O)CN(C(c2cnc(O)c(Cl)c2)=O)C1 CCC(C(=O)NC(C1CCCC1)CNC(c1ccc(C2CC2)nn1)=O)C(F)(F)F C1(CCCNC=O)CCCCN1C(=O)CC1CCCC12CC2.C1(CO)(CO)CCC1 C1(NC(c2c(C)con2)=O)(CO)CCN(CCOC2CCC2)CC1 N1(C(C(C)c2cccs2)=O)CCC2(CNC(C3(CO)CCC3)=O)CCCC12 N1(C(c2c(C)ccnc2O)=O)CCCN(C(=O)CCOC2CCCCC2)CCC1 N1(C(CC2(C)CNC2)=O)CCCc2c(CCN)cccc21 c1(C(N2CC(c3cn(CC(CC)O)nn3)(O)C2)C2CCCC2)ncccc1Br C1(NC(C(C)(C)CF)=O)CC1C1CCN(C(C2CC(=O)CCO2)=O)CC1 CC(C)C#CC(=O)N(C(C)CNC(c1ccc(-c2ncon2)cc1)=O)C CCCC(C)(O)C(=O)NC1CC(C)N(C(=O)CCNC(=O)C(C)(C)C)C1 c1(CN(C2CN(C(c3ccc(O)cc3)=O)C2)C)cc(OC(F)(F)F)ccc1O c1(C(=O)NC2C(C(=O)NC(C(=O)OC)CO)C2(C)C)cccc(F)c1 CC(C)C(C)(C)C(=O)N1CCOCC(C(=O)NC(c2nccc(O)n2)C)C1 C(c1c2c(nn1C)CCCC2)=CC(=O)NC(C(=O)OC)(C)Cc1cccnc1 c1(COC)nc(OC)cc(NC(C2CCCC2)CNC(=O)CC(C)O)n1 c1(C(=O)NCC(n2cc(CN3CCCCCC3)nn2)C)cc2c(Br)coc2cn1 N(C1COc2cc(Br)ccc21)C(c1n(C(C)C)nnn1)(C)CCI C(=O)(C1c2c[nH]nc2CN1C(=O)CC1=CCCCC1)N(CC(C)C)CCO c1(CCNCC2C(Cl)(Cl)C2)ccc2c(c1)OC(F)(F)O2 C1(NC(C(CC)SC)=O)CN(C(=O)Cc2nc[nH]n2)CCC12CCOCC2 C1(C(=O)NCC#CC(=O)NCCC(=O)OC(C)=O)(OC)CCC(C)C1 c1(C(=O)NCCNC(C(C2CC2)SC)=O)cncc(F)c1Cl.C12(CC1(F)F)CN2 c1(C(N2CCC(CC#C)(C(=O)NC3CN(CC)C3)C2)=O)ccnc(C)c1C C1(OC(c2csc(-c3cccnc3)n2)=O)CCCC2CCOC12 C1(NC(c2c(C)ccnc2)=O)CCN(c2ccc(C(F)(F)F)cn2)CC1F C=C1CCN(C(c2cocc2C)=O)C(C(=O)NCC=CC)C1 N1(C(CCC#CC)=O)CC2(CCC2NC(c2nc(C)ncc2Cl)=O)C1 CCCCC(C(=O)NCCCCCNC(C1CC2CC2(CC)C1)=O)C(C)C Cc1ccc(C(=O)NC23CCN(C(=O)CSCC(N)=O)CC2C3)c(O)n1 C(=O)(C1=CCCN(C(c2cc(C)c(N)cn2)=O)C1)NC(C1CCCCC1)CC c1(C(=O)NCC(CC(C)C)NC(=O)Cc2nc[nH]n2)c[nH]c2ncccc12 CCC(C(=O)N1CC(O)(CNC(=O)CSC2CCOC2=O)C1)C(F)(F)F c1(C(N2CC(N(C(C3CCC(CC)C3)=O)C)C2)=O)cn(C)nc1-c1ccoc1 C1(NC(C2(F)C(C)C2)=O)CN(C(c2onc3c2CCCC3)=O)C2(CCC2)C1 C=CC1(OCC(N2CCC(C)C2CC)=O)CCOCC1.N12CCC(C1)C2=O c1(OC)nc(Cl)c(C(=O)NCC(C)(C)CNC(=O)Cc2nncn2C)s1 c1(COC)csc(CN2CCC(N(CC(O)Cc3ccccc3)C)C2)c1 N1(C(C(C)C)=O)CCN(C(=O)CC(F)(F)Br)C(C2CC2)C1 c12ccc(cc1)CNC2c1n(CC(=C)C)nnn1.c1(CSCC)ccc(OCF)cc1 c1(C(N2C(C)(CNC(=O)CC=C(Cl)Cl)CCC2)=O)cnc(O)c2ccccc12 c1(C(=O)NCC2(O)CN(C(=O)CCCC3CC3)C2)ccc(F)c2cccnc12 C(C(O)CC(=O)N1CCCC1CNC(=O)CC1CC12CC2)N(C)C C(=O)(CC(C)(C)OCC)NCCCC(=O)NC(COC)CCO CC(CC(N)=O)C(=O)NCC1COCCN1C(=O)CCC1(C)CC1(F)F c1(C(C)C)ccc(C(=O)N(C2C3CN(C(c4ccc(=N)[nH]c4)=O)CC23)C)cc1Cl N1(C(C23CC(NC(c4[nH]cc(C)c4C)=O)C(OC2)C3)=O)CCC2CCCC2CC1 C(C(COC)CC(=O)N1CC(CNC(=O)CC2CCCC(C3CC3)O2)C1)OC C(=O)(C1=CC2(CN(C(C3OC4CCC3C4)=O)C2)OC1)NC(C)Cc1nn[nH]n1 C1(NC(CC(C)c2ccccc2)=O)CC2CC(NC(C3CCC3)=O)C2C1 Cc1ccc(Oc2ccc(C(=O)NCC(C)NC(c3cnn(C)n3)=O)nc2)cc1 N1(NCc2ncc(C)s2)CCN(C(c2cccc(CCO)c2)=O)CC1C(F)(F)F C(C(C(=O)NCC(O)CN(C(=O)CCC(=O)NC1CC1)C)C(C)(C)C)OCC=C c1(C(=O)NC2C(NC(c3c(CC)c[nH]c3)=O)CCC2)cccc2c1C(C#N)C2 C(CCCCCNC(C1(F)C2CCCC12)=O)N(C(=O)CC1(CO)CCCC1)CC c1(CC)nc(C)c(C(=O)NC(C)C(C)NC(=O)C(c2cccc(F)c2)(C)C)o1 c1(N2CC(C)(C)CC2=O)nc2ccccc2s1.Cc1cnn(C2CC2)c1C(=O)O CCC(C)(C)CC(=O)NC1COCCN(C(c2nc(Br)cnc2N)=O)C1 C1(CNC(C(c2cccnc2)OC)=O)CCOC1C(=O)NCC1CC(F)(CO)C1 CCCC(C(=O)NCCCN(C)C1CC1)NC(c1snc(O)c1Cl)=O c1(C(N2CC(CNC(c3c(OC)nsc3)=O)C(C)C2)=O)ccc(F)cc1C CC1CN(C(C2(C)CCCN2C)=O)CC1NC(c1coc(C(F)F)n1)=O c1(CC(=O)NCC(C)N(C(=O)C=Cc2ccco2)CC)ccc(C)cn1 C=CCCN=C(NCCN1CCOCC1CC)NC(C)CCC=C(C)C N1(C(CCc2cccc(OCC)c2)=O)CCC(CC)(NC(C2CC2(C)Br)=O)CC1 c1(N2CCC(N(C)C)(C(N)=O)C2)nc(=NCC=C2CCC2)[nH]c2c1SCC2 C1(C(N(CCC)CCNC(=O)C(O)C(F)(F)F)=O)CC(c2ccccn2)=NO1 c1(C(N2C(C(N(C)Cc3ncc[nH]3)=O)CSC2)=O)cccc(F)c1 N1(C(C2C(C)(C)NC(=O)C2)=O)CCC(C2(NC(c3cc(=O)cc(Cl)[nH]3)=O)CC2)C1 CC1CCn2c(C(=O)NOC(=O)C(O)C(C)(C)C)cnc2C1.N12CCCC1C2 C1(C(=O)NCCNC(C2CC2C(F)F)=O)Cc2ccc(F)cc2O1 N1(C(C2CC(C#N)C2)=O)CC2C(CNC(c3cccc(Br)c3)=O)C2C1 N1(C(c2cn(C)nc2)C(=O)NCCN2CCCC2=O)CCS(=N)(=O)CC1 c1(OC)ncccc1NC(=O)C(C1CC1)N(C)C(c1ocnc1C)=O c1(C(N(C)CC2CCCCN2C(C2CC2F)=O)=O)c(F)cncc1Cl C=CC(C)(O)CC(=O)NCCCCC(=O)NC(C)CCn1cncn1 N1(C(CC(C)CC(C)(C)C)=O)CCc2ccc(F)c(F)c2C1 N1(C(Cc2ccn(C(C)C)n2)=O)CCN(C(C2CN(C)CC(C)O2)=O)CC(O)C1 C1(C(=O)OCC(=O)NC23CC(C)(OCC2)C3)CC2CC3(CC3)CC2C1 CCC(C)(CO)C(=O)NCC1CC(O)CN1C(=O)CCC(=O)c1ccc(Cl)cn1 n1(CC=C)c(N2CCN(CCC#N)CC2)nnc1C1CCCS1 C1(N(C2CCN(C(=O)COCC(F)F)C2)C)CCCN(C(=O)C(=O)N(C)C)C1 C(=O)(C(C(C)C)n1cnnc1)N(C1CCN(c2snc(CC)n2)C1)CCOC c1(C(=O)NC(C)CNC(=O)COCc2ccccc2)cnc2c(ccn2C)c1 c1(C(=O)NC(C2CCCC2)CNC(C2(C)CC3CC3C2)=O)csc2cccnc12 C1(OC)(CNC(C2CC3(CC3)CO2)=O)CCN(C(=O)C(C(C)C)SC)CC1 C(CC)(C(=O)NCC1CC1CNC(c1cnsc1C)=O)=CCCC C(=O)(C1CCCn2ccnc21)N(c1nnc(C(C)C)n1C1CC(=O)N(C)C1=O)C Cc1ccc(C(=O)N(C2CCCN(C(=O)C(C)OC3CCCC3)C2)C)nc1 C(=O)(C(C)(C)CCNC(=O)Cc1cccs1)NC(CCC)C(=O)NC N1(C(CCC2C(C)C2)=O)CC2CCC(C1)C(NC(C1CC1C1CCC1)=O)C2 c1(C(C)(C)OC)nc(C)c(C(=O)NCC2CN(C(C3CCS3(=O)=O)=O)CC2O)s1 N1(C(c2nc(CCC)sc2)=O)CCCC2(NC(c3nc[nH]c3CC)=O)CC2C1 C1(CC)COCCN(C(=O)C(C)(C2CC2)N(C(=O)C=C2CCOCC2)C)C1 Cc1cccc(CNC(C2CC(O)CN2C(c2cccc(Cl)c2C)=O)=O)c1C c1(C(N(CCNC(=O)C=Cc2nccs2)CC)=O)ccc(C)c(C)c1N c1(C(=O)NC(CCNC(C2(CC)CCOC2)=O)C)c(C(F)(F)F)nn(C)c1C#N C1(NC(C2CN3CCC2CC3)=O)CN(C(C2CC(F)C(=O)N2)=O)CCC1CO N1(C(c2cnc(CC)nc2)=O)CC2(CC(C(=O)NC(C)C(=O)NC(N)=O)CO2)C1 C1(C(=O)NC(C#C)CC2CC2)C(O)CCN1C(=O)Cn1cnnn1 N1(C(C(C)(C)OC(C)C)=O)CCOCC(C)(CNC(=O)CC(C)O)C1 CC1CN(C)CCC1N=c1nc2sccc2c(NCCC2(C)CC2)[nH]1 Cc1nn2ccccc2c1C(N1CCCC(NC(=O)CC2CC(F)C2)C1)=O C1(NC(CCc2onc(CC)n2)=O)CC2CC1N(C(=O)CN(C1CCCC1)C)C2 N1(c2ccnc(C(=O)OC)n2)CCCC(C2CC2NC(=O)C(C)(C)CSC)C1 c1(-c2nc(C(CCC)C)nn2C)ccc(C2CCCN2C)cc1C N(C1CN(C(=O)C(C)CCCOC)Cc2ccccc21)C(C=CC)=O C=C=C(C)CC(=O)NCC1(C)CCCN1C(c1c(Cl)cnn1CC)=O N1(CCC(=O)NC(C(C)NC(COCCCCC)=O)CO)CCCCC1=O c1(C(=O)NCC2N(C(c3c(C)cccc3)=O)CCC2C)cccc(C)c1N C1(C)(C(N(C)CC2N(C(C(C)OCCC#C)=O)CCC2)=O)CCC(=O)N1 c1c2cc(OC)c(OC)cc2oc1.c1(CN(C(C)C(C)C)CC(=O)NC)cccc(Cl)c1 N1(C(C(C(=C)C)(C)C)=O)CCC2CCN(C(c3ccc4cnoc4c3)=O)CC2C1 CC1(C)C(NC(C2CCCC2(F)F)=O)CCN1C(=O)Cc1cccc(C(F)F)c1 c1(CC)ncc(C(N2CCC2C(=O)NC(CO)C2(C)CC2)=O)s1 N1(C(c2n(C)ccc2)=O)CCC2CCN(C(c3ccn4c3CSCC4)=O)CC2C1 c1(C(=O)NC2C(NC(C(c3c(C)nn(C)c3)C)=O)CCC2)cncc2c1CCC2 C1(C(=O)NC2CCCCN(C(c3ccc(CC)nc3)=O)C2)CCCCCS1(=O)=O n1(CC(=O)NCC2CCN(C(C(C3CCCCC3)OC)=O)C2)nc(C)c(C)c1C Cc1cc(C(N2CCCC2C(C)NC(c2snnc2C)=O)=O)cc(Cl)c1 c1(C(N(CCNC(=O)CC2(c3ccon3)CC2)CC)=O)ncnc2c1CCCC2 CC(C)(C)CCC(F)C(=O)NCC1CN(C(=O)Cc2ccc(F)cc2F)CCO1 c1(OC)ccc(C(=O)NCCCc2ccc(Cl)cc2Cl)cc1-c1cccc(F)c1 C1(CNC(C(n2cccn2)C)=O)(CO)CCCN(C(=O)C(O)C2CC2)C1 N1(C(c2sc(CC)c(C)c2)=O)CC(O)C(O)C1CNC(=O)CCCC(=O)N(C)C c1(C(=O)Nc2c(C(=O)OCC)occ2)cn(C2CC2)c2ccc(Cl)cc2c1=O C(C)(C(=O)N1CCN(C(C2(C)CCCOC2)=O)C(C)C1)(C(C)C)NC(C)=O C1(C(C)CO)CCN(C(c2c[nH]nc2CCNC(=O)C=C2CCC2)=O)CC1 C12(CCNC(C=CCOC)=O)CCC(C1)N(C(=O)C(=CC1CCCCC1)F)C2 C(=O)(C1=CC2C=CC1C2)NCC1N(C(C(C=C)C)=O)CC(O)C1 CC1(CO)CN(C(C2COCCN2Cc2ccc(Cl)nn2)=O)CCC1O c1(C(=O)NC2(COC)CCN(C(c3cncn3C)=O)C2)cc2cccc(C)c2o1 c12nn(C)cc1CN1CCC(C1)NC2=O.c1(CC2(CN)CC2)ccccc1 N1(C(c2ncc(CC)nc2)=O)CCN(C(C2(C)CC2Br)=O)C2(CC2)C1 C1(C2(N(C)CCNC(N)=O)CC2)CCCN1C(=O)CC1(C)CCCO1 c1(C(=O)NCCCNC(C2(COC)C=CCC2)=O)cc(C)cc(Cl)c1 C1(C(=O)NCCNC(CCCC(=C)C)=O)C2Cc3cc(Cl)ccc3C12 CC(CN(C)C)CCC(=O)NCC(C)(C1CC1)NC(c1cnc(C(C)(C)C)o1)=O CCCC(CC)CC(=O)NCC1CCN1C(c1cc(CC)nn1C)=O CC(F)(F)CC(=O)NCC(C)(O)CNC(=O)Cn1cc(F)ccc1=O C1(NC(C(C)NC=O)=O)CCCC(C(=O)NC2CCCC(O)C2)CC1 C(=O)(C(CCOC)OC)NC(CCC(N1CCC(COC)CC1)=O)C CC1C(=O)NCCN1C(c1ccc(CNC(C2OCCC2(C)C)=O)o1)=O c1(C(=O)NC(C(C)OC)C(N2CC3(CCCN3C)C2)=O)cc2ncccc2[nH]1 C1(CNC(CCCOCCC)=O)CC(F)(F)CN1C(=O)CCN1CCC(F)C1 Cc1ccc2c(c1)C(CC(=O)NCCN(C(c1ccoc1C)=O)C1CC1)C(=O)N2 C1(C(=O)NCC2(F)CCCN(C(C3CC4(CC4)C3)=O)C2)CCCCC12CCC2 c1(OC)cncnc1C(=O)NC1CC(C(=O)NCCC(F)=C(F)F)C1(C)C C(CNC(=O)COC1CCOCC1)(C(C)C(C)C)NC(c1cnc(C(C)=O)s1)=O C(C(=O)NCC1CC1)(C(C)C1CCC1)N(CCOC)Cc1ccsc1 N1(C(c2c[nH]c(=NC)s2)=O)CC(O)CC1(C)C(=O)NC1(C)CSC1 C(=O)(C1=NOCC1)NCCCN(C(=O)CN(C)C(c1ccccc1)c1cscn1)C C1(NC(CSCCNC(c2cc(C)sc2)=O)=O)CCOC1(C)C c1(CC)ncsc1C(=O)NCCC1(NC(=O)CCC2CC2)CC1 C(=O)(N=c1[nH][nH]c2ccc(F)cc12)NCc1c(C(C)(F)F)cccc1 c1(C(N(C2CN(C(=O)Cc3csc(=N)[nH]3)CC2F)C)=O)cc2c(s1)CN(C)CC2 C1(CNC(C2C(C(C)(C)C)C2)=O)CN(C(c2ccc(F)c(F)c2)=O)CCC1(F)F C12(C(=O)OC)CCC(CNC(C34CC(C(F)F)(C3)C4(C)OC)=O)(CC1)OC2 c1(NCC2(CN(C)C)CC2)nc(NCCCCS(N)(=O)=O)nc2c1ncn2C C1(NC(c2cnc(C)o2)=O)CC(C)N(C(=O)CN(C)Cc2ccccc2Cl)C1 N1(C(c2ccc(CCCC#N)cc2)C(=O)NCCCSC)CCCN(C)CC1C Cc1cc(C(=O)NC2CN(C(c3ccc(OC(F)F)nc3)=O)C3CC23)cc(Cl)c1 C(=O)(CC1=CCN(C)CC1)N1CCC(C(F)F)(CNC(Cc2nc(C)oc2)=O)C1 C1(C(=O)OC)CC2C(CC1C(=O)NCc1ccc(O)c(C)c1)C2(F)F C(C(C(=O)NC1CCCN(O)C1=O)C(C)(C)C)NC(c1c(OC)cccc1)=O N1(C(CNS(NC)(=O)=O)=O)CCC(CNC(c2cccn2C(C)C)=O)C12CC2 CCCC(CC(C)C)C(=O)NCC(CC(=O)NC1CCC(C)(C)CC1)OC C1(C(=O)NC(CC)C(F)(F)F)COC2(C1)CN(C(=O)C(C)(C)CNC(C)=O)C2 N1(C(C=C(C)CNC(=O)COC(C)(C)C)=O)CCC(CCCO)C1 N1(C(C(CCC)O)=O)CCCC12CCCN(C(=O)C(N1CCNC1=O)C)C2 c1(C(=O)NCC(CN(C(CN(C(C)=O)C)=O)C)O)cnc2ccnn2c1C(F)F c1(CC)cc(C)c(C(N2CCCC2C2CCCOC2)=O)o1 c1(-c2nc(NC(=O)COc3nnco3)sc2)cccc(C(F)(F)F)c1.C(C1CC1)N C1(NC(CC(COC)NC(C2CCSCC2)=O)=O)CCN(C)C(=O)C1 C1(SC)CC(NC(=O)COC2CC(NC(=O)CCOC3COC3)C2)C1 C(=O)(C1CCc2scnc21)NC1(CNC(C2(C)N(C)CCC2)=O)CCCCC1 C(C(=O)NOC1CCOC1)(C1(C)CCN1C(C1(F)CCOCC1)=O)CCO C1(C)(CNC(C2C(OC)C2)=O)CN(C(c2cnc(N(C)C)cn2)=O)CC1C Cc1[nH]c(C#N)cc1C(N1CCC(NC(=O)CCC(C)N(C)C)C(F)C1)=O c1(-c2c(CN(C)Cc3ccc(OC)nn3)n(C)nc2)ccc(OC)c(C)c1 S(=O)(=O)(c1cccc(N2C3CCC2CC(=O)NC3)n1)NC(CC)CN1CCCC1 CC1=CC(C(N2CCC2CC(=O)NCC=CBr)=O)SC1 Cc1cc(N2CC3CC2CS3(=O)=O)nc(=NC(C)CCC2CC2)[nH]1 c1(C(=O)NC(CC(C)NC(C(CC2CC2)OC)=O)C)cn(C)nc1C1CC1 N1(C(C(Cc2ccco2)NC(=O)Cc2ccsn2)=O)CCC(F)(F)C(O)C1 CC1CN(C(C2CCCCO2)=O)CCN1C(c1nn(CC(F)(F)F)cc1Cl)=O n1(CC(=O)Nc2n(CC)nc(C)c2)ccc(=NC(=O)CC2CCC2)nc1O c1(C(=O)NCC2(F)CCN(C(C(CC)CC(F)F)=O)C2)nsc2ccc(C)cc12 Cc1nnc2n1CCC(C(=O)NCC1(C)CCCN1C(C1CC3(CC3)CO1)=O)C2 c1(C(=O)NC(C(C)(C)NC(CC(COC)(C)C)=O)C)cc2c(o1)CCCNC2=O C(C)(N=c1ccnc(N2CCC(SC(F)F)C2)[nH]1)c1n(CC)ccn1 c1(C(=O)NCCCC(C)(C)NC(c2cccnn2)=O)cnc2sccn12 C1(N(C(CCN(C(C2C(C)SCCC2)=O)C)=O)C)CCOC(C)(C)C1 c1(C(=O)NCC2N(C(CSC(C)C)=O)CC2)cncnc1C(C)C C1(NC(C=C(CC)CC)=O)C(C)CCN(C(=O)CC2OCCO2)C1C CCC(C)CCCC(=O)N1CCCC1C(C)(C)C(N1CCC([N+](=O)[O-])CC1)=O CC1(CNC(=O)C(C)(C)c2ccccn2)CC(NC(=O)CSC(F)(F)F)C1 N1(CC(=O)NCCC2CC(NC(Cc3cc(C(C)=O)sc3)=O)C2)CCS(=O)CC1 S(=O)(=O)(c1cncc(C#N)c1)NCC(=O)OC(C)(C)C C1(C(=O)NCCc2cccc(Cl)c2)CC12CCN(C(c1cc(Cl)ccc1O)=O)C2 c1(C(=O)NCCCN(C(=O)C(C)CC(F)F)C(C)C)cnc(O)c2cccnc12 N1(C(C2CN(C(CC(CC)C)=O)CC2CC)=O)CC(=O)NCC1CC C12(CC(=O)N(CCc3nccs3)CC)COC(CF)(C1)C2 C1(C(C)C)CN(C(=O)CCOCC(F)(F)F)CCN1C(c1ccc(F)c(Cl)c1)=O c1(CN2CC(NC(C(C)S)=O)C(F)C2)c(Br)ccc(Cl)c1Cl C12(C(=O)NCC3CC[Si](C)(C)C3)CC(CCO1)N(C(=O)CC1CCC(=O)NC1)C2 Cc1nc2ccccn2c1NC(=O)CC1(C)CN(C(c2ncncc2Cl)=O)C1 CCCCC(C(=O)NC1CC2(C(=O)NCC(C)CO)COC1C2)N(C)C N1(CC(=O)NC2CCC(CC(=O)NC3CCCCC3CO)C2)C(=O)CNC1=O CC(C)(C)CCCC(=O)N1CCC(Cn2cc(-c3cnccn3)nn2)C1 CC1(NC(c2cnc(-c3ccccc3)nc2)=O)CCCN(C(c2cocn2)=O)C1 c1(NC(=O)OC)cc(C)c(NC(=O)C(=O)NCc2csc(C#N)c2)cc1C c1(C(=O)NCc2ccc(-c3cnc(C)s3)cc2)ccc(F)c(C(C)C)c1 C1(CCNC(CC(CC)C)=O)CC2CCC(C1)N2C(=O)C#CC1(C(F)(F)F)CC1 Nc1cc(C(=O)NC2CC(NC(C3CN4CCC3CC4)=O)C23CCC3)cc(F)c1 c1(C(=O)NCC(C)N(C(=O)CCCN2CCCC2)CC)ccc2ccnn2c1 Cc1cc2cc(NC(C34COCC3C4(F)F)=O)ccc2o1 S(=O)(=O)(c1ccc(NC2(c3ccc(F)cn3)CC2)c(F)c1)NC1C(C)CCCC1 c1(OC)cc(Br)ccc1C(=O)C(=O)NCC1CN(C(=O)CCC2CCC2)C1 Cc1cc(C(=O)NCc2nc(CNC(C3C4CC5C(C4)C35)=O)cs2)sc1C c1(CC(=O)NC2(CC=C)CN(C(C3CSCCS3)=O)C2)c[nH]c2cc(F)ccc12 C1(C(=O)NCCC(C)CCNC(C2CCCN2C2CC2)=O)CC(C(C)(C)C)=NO1 CCCC(C)(CC)C(=O)NCCCCN(C(=O)CC(C)N1CCCC1=O)C N1(C(C(C)NC(CC)=O)=O)CCOCC(F)(CNC(c2nn(C)cc2SC)=O)C1 N1(C(C(CC=C)CC=C)=O)CCC2CN(C(=O)COCC3CCCO3)CCC12 c1(C(N(CCCCN(C(=O)CCCCNC(N)=O)C)C)=O)cccn2nccc12 N1(C(CCn2c(C)ncc2)=O)CCC2CCC(C1)N2C(c1ncoc1C(C)C)=O c1(C(=O)NC2C(C)N(C(=O)Cc3cncc(C#N)c3)CC2)cc(O)cc(O)n1 CC1CCN(c2cc(NCc3ncoc3C(F)(F)F)ncn2)CCS1 c1(CC(C(=O)O)NC(c2ccc(C(=O)OC)cn2)C)ccc(Br)c(F)c1 C1(C(=O)O)CC12CCCCC2.C1(CN(CC)CC)CCCN1C(=O)C1CC1 C1(NC(CC(CC)(F)F)=O)CCC(O)CN(C(=O)Cc2c(F)cccc2F)C1 N1(C(C(C)(C)OC)=O)CC2(C(=O)NCCC34CC(CCO3)C4)CCC1CC2 c1(C(N2CCN(C(c3c(CC)occ3)=O)C(C)C2C)=O)c(C)cc(C#N)cc1C N1(Cc2cnc(C(C)C)nc2)CCC2CC(C(=O)NCc3ccc(O)nc3)C2C1 Cc1ccc(C(=O)N(CCCNC(=O)C(C)NC(=O)C(F)(F)F)C(C)C)o1 C1(c2n(CCOCC)nnn2)(NCc2ncccc2Cl)CCC(CC)C1 S(=O)(=O)(c1ccc(F)c(Br)c1)N1C2CN(C(c3cncnc3)=O)CC21 N1(C(C(C)(C)C2(O)CCC2)=O)CC2(CC(CNC(=O)C3=CCCCCC3)CO2)C1 C1(C)(C(=O)NCCCN(C(=O)C(C(C)C)n2cnnc2)CC)CCCCNC1=O Cc1cc(F)sc1C(=O)NCC(C1CCOC1)NC(c1ccncc1N)=O c1(-c2n(CCCN(C)C)nc(COC(F)(F)F)n2)cccc2ccncc12 C1(CNC(C(C)=C2CC2)=O)CCC2(CN(C(c3cnc4n3CCCC4)=O)C2)O1 N1(C(C(CSC)C)=O)CCC2CCN(C(C3CCC(C)CC3)=O)CC2C1 C=CC1(CC(=O)NC2CCCC(CN(C)C(c3cscc3C)=O)C2)CCCCC1 N1(C(CC(C)N(C(CCCSC)=O)C)=O)CC2(C1)CC1(CCC1)C2 Cc1c(C=CC(=O)NCCOC2CCN(C(C3(C)CC3(C)C)=O)C2)cnn1C CN1CCC(C(=O)NCCc2ocnc2CNC(C2CNC(=O)C2)=O)C1 CCC(CC(=O)NCC1(NC(=O)C(C)(CC)OC)CCC1)C(C)C CN=c1[nH]cc(C(N2CCCC2(C)CCC(=O)NCC(O)C(N)=O)=O)s1 C1(N(C(=O)CCc2ccon2)CC)CCCN(C(=O)CCn2nc(C)cc2C)C1 C1(C(N2CC(NC(c3sccc3Cl)=O)C(CC3CC3)C2)=O)CCCC12CCC2 C1(C(N(C(C(N2CC(C(=O)NC)C2)=O)C)C)=O)CCCCC1C(N)=O N1(C(CC(C(C)OC)NC(COCCCOC)=O)=O)CC(CO)CC12CCC2 c1(C(=O)NCC23C(CN(C(C4(COC)CCCO4)=O)C2)C3)occ2c1CCOC2 c1(COC)cc[nH]c1C(=O)NC(C)(C)C(=O)Nc1cccnc1 c1(C(N2CC(C(=O)NCCCOC)NCC2)=O)ccc2c(Br)nn(C)c2c1 C(=O)(C1=NN2CCCN=C2N1)NCCCC(C)(C)NC(c1n[nH]cc1Br)=O CC#CC1CN(C(=O)CN(C(=O)Cc2ccc(C)o2)C(C)C)C1 Cc1cc2[nH]c(C(=O)NC(C)CN(C)C(C3CCCC(O)C3)=O)cc2o1 c1(NC(C2(O)CCN(C(c3nn(C)c(O)c3)=O)C2)=O)cc(Cl)c([N+](=O)[O-])cc1O C1(NC(C=Cc2ccc(C)cn2)=O)CC2CN(C(C3(N(C)C)CCC3)=O)CC2C1 C(C(C(=O)NCC1(F)CC(NC(=O)CCOC)C1)OC(C)=O)OC c1(C(N2CCC(C(C(=O)NCC(C)CN(C)C)(C)C)C2)=O)cncc(F)c1 c1(C(=O)NC(C(C)NC(=O)CSC(F)(F)F)(C)C)nc2ccccn2c1F CC1CC2(CCN(C(C3(C)CCN(C)C3=O)=O)CC2)CN1C(c1cc(Cl)no1)=O Cc1nn(C)c(C(N2CCCC2c2cnn(C)c2)C(=O)NCC2CCCO2)c1Cl c1(OCC)cc(Cl)ccc1C(N1CC2C(NC(=O)C(COC)NC(C)=O)C2C1)=O C(=O)(CCC1=NNC(=O)CC1)NC1CC(CNC(C2(C)C(C)C2)=O)C1 C(=O)(CC(C(F)(F)F)NC(c1ncc(F)cc1N)=O)NC(c1nc(CC)on1)C C1(=CC(N2CCC(NC(C3C(C)OC(C)C3)=O)C2C2CC2)=O)CN2CCC1CC2 N1(C(C2CCC(=O)N2)=O)CCCC(NCc2ncsc2Br)C1 C=CCCC(C(=O)NCCCC1(O)CCC1)NC(=O)CNC1CCCC1 CCCCC(CC)C(=O)NCc1ccc(C(=O)NCCC(C)N2CCCC2)cn1 C1(O)(C(=O)NCC(C)NC(c2cccc(C(N)=O)n2)=O)CCOC1(C)C N1(C(c2cnc(C)n2C)=O)CCCC2(NC(=O)Cc3ccc(F)cc3)CCCC12 C(=O)(C(C)C(C)NC(c1sncc1C)=O)NCC=CCCOC N1(C(C(C2CC2)OC)=O)CCCC(C)(NC(c2c(C(F)(F)F)cccc2Cl)=O)C1 c1(CNC(C2C3CN(c4cc(C(F)(F)F)ncn4)CC23)=O)nccnc1Cl c1(CC)cccc(C(=O)NCC2CCC(NC(=O)CN(C)C(=O)OC)C2)c1N C1(C(=O)NCC2(O)CCN(C(C3(COC)CCC3)=O)C2)CC2CCC(C1)O2 n1(CC(=O)NC2(C)CCN(CC(C)C)CC2)ncc2cccnc12 Cc1nn(CC(F)F)c(C)c1C(N1CC2(NC(c3cncc(F)c3)=O)CC1C2)=O c1(OC)ccc(NC(C2CCCN(S(=O)(=O)CC(=O)O)C2)=O)cc1Br C1(C)(C(N(C2CN(CC(=O)NCc3ccccc3)C2)C)=O)CC1(F)F c1(CCC)ccc(C(=O)NCC2CCCC2NC(C2(COC(C)C)CC2)=O)cc1 C1(CNC(CSC)=O)CCC2(CN(C(=O)CCOc3ccccc3C)C2)O1 Nc1cc(Cl)nc(C(=O)NC2CCN(C(c3nncn3C3CC3)=O)CC2)c1Cl C(N=c1[nH]c(N2CCCC(c3cc[nH]n3)C2)nc2c1SCC2)C1(OCC)CCC1 N1(C(C2N(C)C(=O)CC2)=O)CCCC2(C1)CN(C(c1cncn1C(F)(F)F)=O)C2 Cc1ccc(C(N(CCN(C(=O)C=CCC2CC2)C)C)C)o1.C(C(F)(F)F)N CCCCCCCN(C)C(C1CC(n2cc(CC3(O)CCSC3)nn2)C1)=O C12(C(=O)NCC3CCC(C)C3)CC(CN(C(=O)C(F)F)C1)C2 c1(C(=O)NC2CCN(C(C3C(C)OCCO3)=O)C2)c(F)ccc(F)c1Br c1(C(C)(C)C)ncc(C(=O)NC(C2CCOC2)CNC(=O)Cc2cn[nH]c2)o1 C1(C(=O)NCC2(C)CC(C)(C)C2)(CC)CCCN(C(=O)C(F)=C(C)C)C1 Cc1cc(NC(C2(NC(=O)C(C)C(F)F)CCC(C)(C)C2)=O)cc(O)c1 C=CC(C)(C)C(=O)NC(CN(C)C(c1cc(-c2ccns2)on1)=O)CC N1(C(c2ccc(NC)cn2)=O)CCCC(NC(c2cn(C(C)C)cn2)=O)CC1 CC(C)C(CNC(c1n[nH]c(=N)[nH]1)=O)C(=O)NC1(CO)CC2CCCC12 N1(C(c2cnc(OC)s2)=O)CCCC2C1CCN2C(=O)Cn1nc(C)oc1=O C12(C(N3CC(CC(C)C)OCC3)=O)C(NC(c3ccc[nH]3)=O)C3CC1C2C3 c1(C(=O)NOC(c2ccc(CO)o2)=O)ncoc1CSC1CC1 O=C(Cc1cnc(COC(F)(F)Cl)o1)NNC(=O)c1ccccc1 c1(C(CC(C)C)NC(=O)C(=O)Nc2ccc(Br)cc2)ccc(F)cc1 C(CC(=O)N1Cc2ccccc2CO1)(c1ccccc1)OCCOC CC1CN(C(=O)CCCc2cccc(Cl)c2)CC(C)N(C(=O)COCCO)C1 N1(C(c2ccc(OC)o2)=O)CCCC2(CCCCC2NC(c2oncc2C)=O)C1 c1(C2N(C(N(C(C3CCC(C)O3)=O)C)=O)CC2)ccccc1Cl.C1(CN)(C)CCC1 C1(NC(C2(CC)CCOCC2)=O)CCC2CC1CN2C(C1CCC(CC)CC1)=O C1(=O)C(F)(F)CCC(=O)N2C(CC2)CN1.CC1(F)CC(C(=O)OC(C)(C)C)C1 C(=O)(C(O)CC(C)(C)C)NCC(CNC(c1cnc(C(C)O)s1)=O)(C)F N1(C(C(c2ccc(C)cc2)=O)C)CCC2C(C1)NC(=O)N2C c1(CC(=O)NC2CC23CC(NC(C2(O)CC2)=O)C3)c[nH]ccc1=O c1(C(C(=O)NCCCSC)N(C)CC2CCOC2(C)C)sc(Br)cc1C C12(CC(=O)NCCOC3CCN(C(C(C)C4CC4)=O)C3)COC(COC)(C1)C2 CC(C)(CC1CC1)C(=O)NCC1C2CC1N(C(c1ocnc1C(F)F)=O)C2 C1(C(=O)NC2(C)CC(NC(C3CN(C(C)C)C(=O)C3)=O)C2)OCCN(C)C1=O C1(NC(c2c(C)noc2)=O)CCN(C(c2sc(-c3ncc[nH]3)nc2C)=O)CC1F N1(C(C2CSCCS2)=O)C2CCCC1CN(C(=O)C(F)(F)c1ncccn1)C2 N1(C(=O)C(O)Cn2cncn2)CC2CC1CN2C(C1(c2cccc(F)c2)CC1)=O C(CCCCCC(=O)N1CCC(O)(CN(C(=O)CN2CCC(C)(C)C2)C)C1)SC N1(C(C(CCOC)(C)C)=O)CCN(C(C23CCC(CC2)C3(C)C)=O)CC(O)C1 c1(C(C)C(=O)NCc2nc(-c3cccs3)n[nH]2)ccc(F)cc1F Cc1cc(C(=O)NCC2(C(=O)NC3CCN(CCCO)C3)CC2)cc(O)n1 C(N=c1ccnc(N2CCOCC(F)(F)C2)[nH]1)C1CCCC(C)O1 C1(N(C(C(N2CC(C)C2)C)=O)C)CCCN(C(c2nn[nH]c2Cl)=O)CC1 Cc1cc(C(=O)NCC2(C)CCCN2C(C2CC=CCO2)=O)cn(C)c1=O C(=O)(C1=C(Cl)CCCC1)NC(C(C)OC)C(=O)N1C2CCC1CC2 C1(NC(CCCCNC(N)=O)=O)CCN(C(=O)CC2=CCCC2)CC12CCC2 C1(CCNC(CSc2n[nH]c(=N)s2)=O)CCN(C(=O)CC2(O)CCOCC2)CC1 CC1(C)CN(C(C2CCOCC23CCC3)=O)CC(CNC(=O)CN2CC=CC2)O1 c1(C(NOCC(=O)N(CCCO)CC)=O)cc(C)c(C)nn1 S1(=O)(=O)c2ccc(C)c(c2)N(CCOC(C)=O)N1C.c1(NC)cccc(Br)c1 C1(N(C(C(C)Cn2cccn2)=O)CCNC(C2(C(F)F)CC2)=O)CCCCCC1 N1(C(c2ncccc2F)=O)CCCC(N=c2nn[nH]n2-c2ccccc2)C1 C12(C(=O)NCC(C)N(C(c3cc(F)ccc3F)=O)CC)CCCCC1OCC2 C(C(C(=O)NCC1CC1(C)C)N(C)C)NC(C(C1CCC1)OC)=O C1(NC(c2cnc(Cl)s2)=O)C2CC1CN(C(C1CC3C(C1)C3(F)F)=O)C2 C(=O)(N=c1[nH][nH]c2c1CN(C(c1ccc(Cl)c(I)c1)=O)C2)c1ccc(C)c(F)c1 C(=O)(CCCC(F)(F)F)NCCC(C)(C)C(=O)Nc1cccc(OCF)c1 O=S(=O)(c1cccnc1NCCC1CC1C1CC1)NCCCN1CCSCC1 N1(c2ncnc(C)c2F)CCC2(CCN(C(=O)Cc3c(F)cncc3Cl)C2)C1 C(CCCCC(=O)NC1CCN(C(c2cccc(C#N)n2)=O)CC1F)N(C)C N=c1[nH]c(C2CC2)ncc1C(N1CC=CC1CNC(=O)CCC1CCOC1)=O N1(C(CCC=CCC=C)=O)CCCCC(CNC(=O)Cc2cc(Cl)sc2Cl)C1 CC1CC(C(N2CCC(OCCNC(c3c[nH]c(Br)c3)=O)C2)=O)CCS1(=O)=O N1(C(C2(F)CN(C(c3c(N)non3)=O)C2)=O)CC2(CCC1CO)CC2 N1(C(C2C(OC)CCCC2)=O)CC2CCC(C1)N2C(C1CC(C#N)C1)=O C=C(C)CC(C(=O)Nc1ccc(C(F)(F)F)cc1SC)NC(C1CCCC1)=O C12(CNC(CC)=O)CN(C(c3cn(-c4cnn(C)c4)cn3)=O)CC1CCO2 CC1C(NC(c2ccnc(C3CC3)c2)=O)CCN1C(=O)C(F)C1CCOC1 C(C(C)(C(=O)NOCC1(C)CCC1)NC(=O)C(C)c1cc[nH]n1)SC CC(C)CC(C(=O)N1CCOCC(C(=O)N(C)C)C1)NC(=O)C(=O)NC(C)(C)C C(=O)(CC(C)(C)C(=O)NCC1CC(OC)CN1C(C12CSCC1C2)=O)OC C1(NC(N(C)C2CC2)=O)CNC(=O)CN1C(C1CC1C(F)(F)F)=O Cn1ccc(CCNC(=O)CC2CC2CNC(C2CC2Cl)=O)n1 CCC(CCCC(=O)N(CC(F)F)CC(C)O)NC(=O)C(C)CC O=C1CC(=O)CC(C(=O)N(CCC(=O)NC2CCN3CCCC23)CC2CC2)C1 c1(NC(C)=O)ccc(F)c(C(=O)NC2CCCCC2CNC(=O)CC#N)c1 CCCCCC(O)C(=O)NC1CCCC(C(N2CC(C3CC3)(COC)C2)=O)C1 CC1CC(=O)CCC1C(=O)N(CC(C)(C)CNC(C12CC3CC1C2C3)=O)C Fc1ccccc1CNC(=NCC1CC1(Cl)Cl)NC1CCOCC1 c1(C(=O)Nc2c(C(C)=O)cc(F)c(F)c2)c[nH]c2cc(C3=CCSCC3)ccc12 N1(C(c2cc(C(C)C)no2)=O)CC(C(=O)NCC(C)N(C)C)C2(CC2)C1 O(NC(=O)C(c1ccco1)NC(c1cccn1C(C)C)=O)CCCC(=O)OC C(N=c1[nH]c(N2CCOC(C(N)=O)C2)nc(=N)[nH]1)c1ccc(NCC(C)C)cc1 N1(C(C#CC(CNC(CC=C(C)C)=O)(C)C)=O)CCC2(CC1)CN(C)C2 C1(CNC(C2CCCN(CC)C2)=O)CN(C)CCN1C(C1OCCO1)=O C1(C(=O)NC2CCN(C(=O)C=C(Cl)Cl)CC2CO)Cc2ccccc2CO1 N1(C(CCSCCC)=O)CC2CC(NC(=O)CCC=CC(C)C)CC2C1 c1(C(N2C3(CNC(C4(NC(C)C)CC4)=O)CCC3CC2)=O)coc2ccccc12 Cc1cnc(C)c(NC(C2C3CCC(C3)N2C(=O)CCC2CCOC2)=O)n1 CC1(C(N2CCC(C(CO)NC(=O)C=C3CCC3)CC2)=O)CC2CC2C1 C1(OCC)CC2(C1)CC2C1CCN(CCCC(=O)NC)C1.c12sccc1OC2 C(=O)(CN=S(C)(C)=O)NCC1CC(OC)CN1C(C1CCCN(C(C)C)C1)=O N1(C(C=CC(CC)C)=O)CCC(CN(C(=O)CN2CCCNC2=O)C)CC1 N1(C(C(C(C)C)F)=O)CCCN(C(=O)CC2CC2)CC1C C(C(C)(C)C(=O)N(C)CC1CCN(C(c2ccc(C3CCOC3)cc2)=O)C1)OC C1(NC(CCOCCOCC)=O)CCCCCN(C(=O)C2=CCCC2C)C1 Cc1[nH]ccc1C(=O)NCC(Cc1ccccc1)NC(=O)CC1C=CCC1 C1(C(=O)Nc2c(C)csc2)CN(C(=O)CCc2cn[nH]c2)CC1C CCCCC(O)C(=O)NC(C)(C)CNC(c1cc(C(F)F)cs1)=O CC1(C)CCC(CC(N2CCC(C(C)(C)C#N)CC2)C(=O)NC2CCC2)C1 c1(NC(Cc2ccc(C(CC(C)C)=O)s2)=O)cn2c(n1)CC(OC(C)(C)C)CC2 C1(OC)CCC2(C(N3CC(CCNC(=O)CS(=O)(=O)NC4CC4)C3)=O)CC12 c1(C(=O)NCCCN(C(C(CCC)C)=O)C2CC2)c(C)oc(C)c1C C1(C(=O)NC(COCCCNC(C(C2CC2)SC)=O)(C)C)CC2CC1CC2(F)F C(=O)(CC(C)CC(F)(F)F)NCCOCCNC(C(C1CCCC1)OCC)=O C1(CN(CC(F)F)CCOCC)CCCC(C(F)(F)F)O1 c1(CNC2C(C)CN(C(=O)OC(C)(C)C)C2)oc2ccccc2c1C(F)F C(c1cccc(OC)c1)=CC(=O)NC(CNC(c1ccc(CC)cn1)=O)CO Cc1ccc(C(N2CC3CCC3(NC(=O)CN=S(C)(C)=O)C2)=O)c(C2CC2)c1 N(C(=NCC(C)N(C)C)NC(c1cccc(Cl)c1)C)C(C=C)C Cc1ccc(NC(=O)C(C)(C)NC(=O)CC2CCC(=O)C2)c(O)n1 Cc1nn(C)c(C)c1CC(N1CCC(NC(c2cccc(=O)o2)=O)C(O)C1)=O C1(CC(=O)Nc2cccc(OCC(F)F)c2)COC2(CCC2)CO1 Cc1ncc(CCC(=O)N(C(C)CNC(=O)C(O)c2ccsc2)C)s1 C12(CNC(c3cnc(S)[nH]3)=O)CCCC1CCN2C(c1coc(C(F)(F)F)c1)=O N1(C(c2c(C(C)C)scn2)=O)CC(CNC(C2CCC(=O)NC2)=O)C(C)(C)C1 c1(C(=O)OC)ccc(NNC(=O)N=c2[nH]nc(CCC(C)C)s2)cc1F CC1(C)CN(C(=O)CN(C2CCC2)C(C2CC2[N+](=O)[O-])=O)CC1CO c1(C(N(C2CCN(C(C3CC(F)C3)=O)CC2)CCC)=O)ccc2nc(O)[nH]c2c1 c1(C(N(C2CCN(C(=O)C=C3CCOCC3)C2)CCC)=O)ccn2c1CSCC2 c1(C(=O)NC(CCNC(CCCNC(C)=O)=O)C)ncn2c1CCC2 C1(N(C(CNC(CCC)=O)=O)C)CCCCN(C(=O)C(C)=C(C)C)C1 N(C(=NCCCC1CC1Cl)NCC1CC1)CC(c1c(C)nn(C)c1C)O CC(CC(=O)NCC(C1CC1)N(C(=O)CC1CC(C)CC(C)(C)C1)C)C(C)(C)C N1(C(C(CC)n2cccn2)=O)CCC(C(CO)NC(=O)CN(C)CC)CC1 C1(CC=C)(NC(=O)C(C)CC)CCCN(C(=O)CC(=O)OCC)C1 N1(C(C(C2CN(C(=O)CC3CC=CCC3)C2)OC)=O)CCCOCC1C c1(NCc2cn(C)nc2)cc(-c2ccnn2C2COC2)ccn1 c1(C(N2CC(O)CC(NC(CCCOCCC)=O)C2)=O)ccc2ncn(C)c2n1 CC(C)(CNC(c1cnc(S)nc1)=O)CC(=O)NCC1(O)CC1 Cc1cccc(CN(CCc2ccccc2)C(C2CCN(C)C2=O)=O)c1 C(C(C)(C)CC(C)C)NC(C=CC1N(C(CC(=O)OCC)=O)CCC1)=O C1(COC)(COC)CC1C(=O)N1CCCCC1.c1(C(=O)NCC)cnco1 CCC(CC(F)F)C(=O)N(CCCCN(C)C(C1C=C1C)=O)C c1(C(c2n(CC=C)nnn2)NC2CC(=O)N(O)C2)nc(C)c(C)n1C C(=O)(C(=O)N=c1cc(C)o[nH]1)N1C(C)CC2CN(C(C(C)OCC)=O)CC21 CN1CC2CCN(C(C34CCC(NC(=O)CCCC#N)(CC3)C4)=O)C2C1 Cc1ccncc1CC(N1CCC(CNC(=O)C(O)C2CC2)C1)=O C1(NC(c2cnc(C3CCC3)s2)=O)C=CCN(C(C2(CCF)CCOCC2)=O)C1 CCCC(CCC)=CC(=O)NC1CCOC1C(=O)NCC1CC(F)(F)CO1 c1(SC)cc(C(=O)NC(C)(CNC(=O)C(C)(O)c2ccccc2)C(C)C)c(C)o1 C(=O)(C(CCCC)SC)NCC(CCCC)NC(=O)C(C)(C)COCC CCC(CCC(=O)N(C)CCc1cnc[nH]1)NC(=O)CSC1CC1 C1(NC(c2cc(OC)c(C(N)=O)cc2)=O)COC2C(NC(=O)CC(C)F)COC12 c1(SCC(C)N(c2n(CC)nnn2)C)ccnc(OC)c1Br C1(CC)CN(C(c2ccc(CO)o2)C(=O)Nc2ccccc2C)CC(=O)N1 N1(C(Cn2c(C)cc(O)cc2=O)=O)CC2(C)CN(C(=O)C=CCF)CC2(C)C1 C1(CCNC(c2ccc(CCC)cc2)=O)CC(F)(F)CN1C(=O)CCCN(C)C C(=O)(C(C)C(O)C(C)C)NC(CC)(C)CNC(=O)Cc1ccccc1 c1(C(N2CCCC2C#N)C(=O)NC(c2ccccc2)C)ccc(OCC#N)cc1 N1(C(CC(C)OC)=O)CCOc2ccccc2C1CO Cc1ccc2n[nH]cc2c1C(=O)NCC1CCN(C(=O)C(C)O)CC1(F)F C=CC1(C(N2CC3CC(F)CC3C2)=O)CCN(C(c2cccnc2C)=O)CC1 C(c1c(F)ccc(Cl)c1F)=CC(N1CC(N(C(=O)C(O)Cn2cncn2)C)C1)=O c1(OC)ccc(C)cc1CN1CCC1CNC(c1cnc(C(C)(C)C)cn1)=O c1(COC)nc(C(=O)NCCOCCN(C2(n3ccnn3)CC2)C)cs1 C1(C(N(CC(CNC(c2c(CC)cno2)=O)C)C)=O)CC2CCCC(C1)C2(F)F C1(C2CN(C(c3ccnc(-c4ccco4)c3)=O)C2)(NC(c2c(C)[nH]cc2)=O)CC1 C(=O)(CC(C)OC)NCC(=O)NCC(=O)NCC=C CCC(N=c1[nH]c(N(C)CCc2nccs2)nc(=NC)[nH]1)C1CC1(C)C N1(C(c2occ(C)c2)=O)CCC(NC(C2CCC(C)CC2)=O)C2(CCC2)C1 C1(NCC(c2cc(Cl)ccc2Br)O)CCC2(CCCCC2)C1 C(C(C)C)(C(O)C(=O)N1CCC(C(C)(C)NC(c2cccnc2O)=O)C1)OC Cc1cnc(C(N2CCC(C3CCC(C(=O)N(C)C)O3)CC2)=O)cn1 CCCC(C)(C)CC(=O)NCC(C)NC(c1coc(=O)[nH]1)=O N1(C(CC=C)=O)CC(CNC(c2c[nH]ccc2=N)=O)C(C(F)(F)F)C1 N1(C(C=CC(=O)OC(C)(C)C)=O)CCC(NC(c2ccc(CO)cc2)=O)C12CC2 Cc1ccc(C)c(S(=O)(=O)NC2CCN(C(=O)CCC3CC3)CC2O)c1 C(=O)(CC(C)C(C)(C)C)N1CC(CC=C)(NC(C23COCC2C3)=O)C1 c1(CC(C)OC(c2cc(O)ncn2)=O)cccc(Cl)c1 Cc1cccc(S(=O)(=O)NCCC2CCCN(Cc3cc4ccccc4[nH]3)C2)c1 N1(C(C(F)=CCC)=O)CC2(CCC2NC(C2CCC(C(=O)OC)O2)=O)C1 C1(C)(NC(CCC(C)C)=O)CCN(C(c2c[nH]cc2Cc2ccccc2)=O)CC1 c1(NC(C)=O)cccc(C(=O)NCC2CCCN2C(c2csnn2)=O)n1 Cc1nc(CO)sc1C(=O)NCC(C1CCN(C(C2(C)COC(=O)N2)=O)CC1)O c1(C(=O)NC(CNC(CNC(CC)=O)=O)CO)nc2ccccc2nc1C C1(NC(C(n2ccc(C)n2)C)=O)CN(C(=O)C(F)(F)C2CC2)CC(F)(F)C1 O=C(Cc1cccs1)C(=O)NCC1CN(C(=O)CCn2ccnc2)C1 c1(C(=O)NC(CC)CNC(=O)CC2COCC2O)sc(Br)c(C)c1C c1(C(=O)NC(CN(C(C2CC2(Cl)Cl)=O)CC)C)ncc(C(F)(F)F)cc1Cl c1(NC(=O)NC2N(C)c3ccccc3C2)ccc2cc(S(N)(=O)=O)ccc2c1 C1(C(=O)NCC(C)NC(c2c(Cl)ccc(C)c2)=O)Cc2ccc(Cl)cc2C(=O)O1 c1(C(N2CCC3(NC(=O)Cn4ncnn4)C(C2)C3)=O)cc(Cl)cc2cccnc12 C1(C(=O)NC(C2(O)CN(C(C(CCCC)O)=O)C2)C)CN2CCN1C(C)C2 CCCCCNC(C1(CNC(C2CC(F)C2)=O)CCC1)=O c1(N2C(COc3ccc(F)cc3)CCC2)ccc(=O)n(Cc2cn(C)nc2Br)c1 C1(NC(C=CC)=O)CN(C(c2cc(C(F)F)n(C)n2)=O)C(C)(CC)C1 N1(C(C=Cc2cccc(N)c2)=O)CC2CCC(NC(C3(CCF)CC3)=O)CC2C1 C(C(C)(C)C(=O)NCCC1CN(C(=O)Cc2nc(C)sc2C)C1)SC C(=O)(CCS(C)(=O)=O)NCCCCCCN(C(C12CC(OC)C1C2)=O)C n1(CC)nc(C(=O)N(C(C)CN(C(=O)C(C2CC2)OC)C)C)cc1O Cc1ccc(CNC(N2CCC(=Cc3cccc(C#N)c3)CC2)=O)cc1C#N c1(OC)ccc(C(N2CCC(C(C)(C)NC(C3CC(F)(CO)C3)=O)C2)=O)nc1Cl c1(C(=O)NCC(C)CNC(c2cccc3sncc23)=O)cnc2nccn2c1 c1(C(N2CC(N(C(=O)CC3CC34CC4)C)C3(C2)CC3)=O)ccc(Cl)c(F)c1N CC(C(=O)NCC(c1cc(F)cc(Cl)c1)NC(C1(CC#N)COC1)=O)S(C)(=O)=O c1(CCCC)noc(CNC2CCCC2Cc2cncn2C)n1 CC(CCCCNC(=O)C(C)(O)C1CCC1)NC(=O)C(C)(C)CO N1(C2CCN(C(CN(CCOC)C)=O)CC2)C2CCC1CN(C(C1CC1C)=O)C2 C(CCCC(=O)NCC1CC(NC(=O)C(F)CC2CC2)CCO1)N(C)C c1(OC)ccc(C(N2CCC(NC(=O)CC3CCCN3)CC2)=O)cc1N n1(CC)c(C)cc(C(=O)NC2CCN(C(c3ccc(NC(C)C)cc3)=O)C2)c1C C1(NC(CCCOCC)=O)CC2CC(NC(=O)COCP(C)(C)=O)CC12 CN1C(=O)CCC1CC(=O)NC1CCCC1NC(=O)COC1CCCCCC1 Cc1c(C2(C(N3CC(F)(CNC(=O)CC=C(Cl)Cl)C3)=O)CC2)cccc1F CC(C)(CNC(C1CCN1C(C1CN(C2COC2)C1)=O)=O)CCCO N1(C(c2c(OC)nc(C)cn2)=O)CC2CCC1CN2C(=O)CC1OCCC1(C)C C(CC(CC)C(=O)NCC12CC(CO1)N(C(C1(SC)CCC1)=O)C2)=CC c1(CC)[nH]ccc1C(=O)NC12CC(NC(C3CC(C)CO3)=O)(C1)C2 c1(C(=O)OC)coc2cc(C(N3CC(CNC(=O)C(C)C(C)(F)F)C3)=O)[nH]c12 c1(CNC(c2cccc(OC(C)C)c2)C)c(OC)cccc1O c1(OC(C(N2CC(Cn3cc(CC(C(C)C)O)nn3)C2)=O)C)ccc(Cl)c(Cl)c1 Cc1nsc(C(N2CC(CCCCNC(C3(C)CCNC3=O)=O)C2)=O)c1N c1(C(=O)NCC#CCNC(Cn2[nH]c(=N)c(Br)c2)=O)n[nH]c2ccccc12 c1(SCCC(=O)NC2(CC=C)CN(C(c3ncc[nH]c3=O)=O)C2)ccccc1Cl c1(OC)cc(C(=O)N(C(C)CCNC(C2(F)CCCCC2)=O)C)cc(F)c1C#N N1(C(C2(OC(C)=O)CC2)=O)CCN(CCC2CCN(C(=O)C(C)CO)C2)CC1 c1(C(=O)NC2C(CNC(c3nc(COC)[nH]n3)=O)CCC2)cc(C)cnc1C N1(C(c2c(C)nc(CC)s2)=O)CC2CC(O)C1C2NC(C1CCC(=O)NC1)=O c1(CC)sc(C(=O)NC2CN(C(=O)C(C)OC3CCCC3)CC2O)cc1C C1(C(=O)NC(CNC(c2cc(CC)ncn2)=O)C2CCC2)CCC(F)(F)CO1 CC1CC(F)CN1C(C12CC1CCN2C(=O)C(CO)N(C)C)=O N1(C(CC(=C)C)=O)CC2CCC(C1)C2NC(=O)CCCCOCC N1(CC(=O)N(C2CCN(C(C3C(c4ccccc4)C3C)=O)C2)CC)CSCC1=O C(=O)(CC(C)(C)C(C)=O)N1CCC(N(C(CCC(=C)C)=O)C)C(C)C1 N1(C(Cc2c(C)non2)=O)CCOCC1CNC(c1ccc(Cl)[nH]1)=O C(CC(=O)NCC1(F)CCN(C)C1)(C(F)F)NC(c1c(CC)occ1C)=O C#CCC(CC(=O)N1CCC2(CCC2)C1)NC(c1cc(OC)ncn1)=O c1(OC(C)C)cnc(N2CCCC(CNC(=O)C=Cc3nccs3)C2)nc1 N1(C(c2cc(COC)[nH]n2)=O)CCC(NC(=O)CC2CCCC23CC3)C1C1CC1 N1(C(CCN(C)C(C2CCCOCC2)=O)=O)CC(O)CC1C(N)=O C1(C(N(CC(CC)NC(=O)CCCCNC(N)=O)C)=O)CC2CC(O)CC(C1)C2 c1(COC(c2cnc(C3CC3)nc2)=O)noc2ccc(Br)cc12 c1(C(N2CC(C)C(NC(=O)C(C)n3cccn3)C2)=O)cc(Br)ncc1Br Cc1ccc(C(=O)NC(C)C(CO)NC(=O)C(C)n2cnnn2)nc1O C1(NC(C=NOC)=O)C=CCN(C(=O)CC2CC23CC3)C1 c1(C(=O)NCC(C)(O)CNC(C2(Cl)CC2(F)F)=O)nccc2c1CNC2=O N#Cc1nc(=NCCCCCCNC(=O)CSc2ccncc2)cc[nH]1 S(=O)(=O)(c1ccc(O)cn1)NC(CCc1cccc(OC)c1)C N1(C(C(C)SC)=O)CCC2C(NC(=O)CCN3CCOCC3)C12 c1(C(N(CC(CC)NC(CCSCCCC)=O)CC)=O)c[nH]c2c(C)cccc12 N1(C(CC(C=C)C)=O)CCC2CN(C(c3ccc(OCCCC)cc3)=O)CC2C1 N1(C(c2n(CC)nnc2)=O)CCC(NC(=O)C(C)SC(C)C)C12CC2 c1(C(C)C)cc(C(C)(C)NC(C2CC2c2ccccc2)C)n[nH]1 c1(C(N2CCC(N(C)C(C3CCCN3C=O)=O)C2)=O)cc2n(n1)CC(C)(C)CO2 Cc1ccc(O)c(C(=O)NCCC(C)NC(=O)C(C)Cc2ccnn2C)c1 c1(N2CCC(CCN(C)CC)C2)nc(N(CC)CC2CCC2)c2c(ncn2C)n1 c1(CCC(=O)NC2C(CNC(C(C(C)C)CN(C)C)=O)C2)c[nH]c2ccccc12 c1(C(=O)NC2CCC(CC(=O)NCCc3nc(CC)[nH]n3)C2)ccc(C#N)o1 N1(C(C2(C=C)CCC2)=O)CCC(CNC(c2cocc2C(N)=O)=O)(N)CC1 Cc1c(C(=O)NC(CNC(C23CCC(CC2)C3)=O)C2CCC2)c(C(F)F)nn1C N1(C(Cn2c(C)ncc2)=O)CCC2C1CCCN2CC=Cc1ccc(Cl)c(Cl)c1 C(=O)(C1=CCCCCC1)N1CCN(C(C(C)CC2CC2)=O)CC1CC1CC1 C(=O)(C1=CCC(C)CC1)N1CCN(C(C2N(CC)CCOC2)=O)CC1.C1CO1 C1(C(C)NC(C(C)Cn2ccnc2)=O)CCN(C(C2(c3nccs3)CC2)=O)CC1 N1(C(COCC(=O)NC)=O)CCC(CNC(C2(C)CC2C)=O)C(F)(F)CC1 C1(NC(c2n(CC)nnc2)=O)C2CC3C(C2)C13C(=O)NC(C)CN(C)CCOC c1(C(=O)NC(CCCC)CNC(=O)C(C)OCCOCC)ccc2nnnn2c1 CC(CCNC(=O)NC1(C)CCN(Cc2ccccc2)C1)C(F)F N1(C(CCC(=O)NCC)=O)CCCC(O)(CNC(C2CC2C(C)(F)F)=O)CC1 C1(NC(c2cc(C)no2)=O)CN(C(c2cc(C(C)(C)C)no2)=O)CC1C c1(C(N(CCC(C)NC(=O)C2CC2)C)=O)cccc(O)n1 C(=O)(C(C)(C)CC1CCOCC1)NC(C1CCCC1)CNC(C=CC(CC)C)=O N1(C(C2CC(C)(C)O2)=O)CCC2(CCCN(C(=O)COC(F)(F)C(F)(F)F)C2)C1 C1(NC(C(CC(C)C)(C)O)=O)CN(C(=O)C=CC(C)(C)C)CC12CCOCC2 C1(C(=O)NC2CCC(NC(C3(C)CC3(F)Cl)=O)CC2)CC2C=CC1C21CC1 N1(C(C(C)=C(CC)C)=O)CCC2CN(C(=O)C(C)(C)S(C)(=O)=O)CC2C1 c1(NC(c2cnn(C)c2C2CC2)c2n(CCSC)nnn2)cc(C)cnc1C CC1(C(=O)NCCOC2CCN(C(c3coc(Cl)c3)=O)C2)CCC(=O)N1 C=CCCC(C)N=c1[nH]c(=NCc2cc3c(s2)CCCC3)[nH]c2ccc(Cl)cc12 N1(C(C2(CC=C)COC2)=O)CCC(NC(c2cccc(OC)c2)=O)C(F)C1 c1(C(N2CC(N(C(C(C(C)C)NC(=O)OC)=O)C)C2)=O)cnc2nccnc2c1 c1(C(=O)NC2CCC(NC(c3c(C)cc[nH]c3=N)=O)C2)coc2c(F)cccc12 CCC(C)C(O)C(C)C(=O)NC1(C2CCCN2C(=O)CCCC2CCC2)CC1 C1(NC(CCSC)=O)CCCN(C(c2ccc(C(C)(C)C)cc2)=O)C1C C1(NC(C2C(=C)C2C(=O)OC)=O)CC(NC(=O)C(C)c2cc[nH]n2)C(O)C1 c1(C(N2C(CC(C)O)CCCCC2)=O)nnn2c1COCC2 CC(C(C)(C)O)N(C(=O)CN(C(=O)CC1CCCN1C)C1CCC1)C C1(C(N(CC(CC)NC(=O)CNC(c2ccncc2)=O)C)=O)(OC)CCSC1 N1(C(=O)NCC2(C(C)(C)C)CCCCC2)CCC(C(F)(F)F)C(CN)C1 c1(C(=O)NCC2C(C(=O)NCC3(C)CNC(=O)O3)OCC2)cccc(C#N)c1 C(C)(CC(=O)NC(C1(CNC(=O)CCOCC2CCC2)CC1)C)SC CC1CN(C(=O)CCNC(=O)CCN(C)C)CCC1NC(C1CCCN(C)C1)=O c1(C(=O)NCC2(F)CN(C(C3CC(C)NC(=O)C3)=O)C2)cnn2c1CC(C)CC2 C1(CNC(Cn2nnc(C)n2)=O)CCC12CCN(C(=O)CC1CCCC1O)CC2 C(=O)(CCC(C)CN(C)C)NC(C(=O)NC(C)C(C)(C)CO)C1CCC1 N1(C(C)C)CCc2onc(C(=O)NCCN3CCCN(C(=O)CNC=O)CC3)c2C1 c1(C(=O)NC(CCNC(CCCCSC)=O)C(C)C)cc(C)c(C)cc1Cl C(CC(=O)NCC(C)CN(C)C(c1cc(OC)cc(C)n1)=O)(C(C)C)OCC c1(OC)ccc(C(F)F)cc1C(=O)NCC(C1CC1)NC(c1n[nH]c(C)c1Cl)=O C(C)(N=c1nc[nH]cc1C#N)C1OCCN(C(c2ncc(C)nc2)=O)C1 C1(C(=O)NCCC2CC(NC(CCOC(C)=O)=O)C2)CCc2nc(C)ncc2C1 c1(NC(C(CNC(C(CC=C)CC)=O)C)=O)cnc2[nH]cnc2c1 Cc1nc(CC2CC2)oc1C(=O)NCC(C)(F)CNC(=O)CC(C)(C)C N1(C(C(C2CCCO2)NC(c2ccncc2)=O)=O)CCOC(CC2CC2)C1 C1(N(C(CNS(CC)(=O)=O)=O)C)CN(C(=O)C(O)c2ccco2)CC12CC2 N1(C(c2c(C)nc(C(C)C)s2)=O)CCN(C(=O)CNC(=O)NC2CC2)C(CF)C1 CC(CSc1ccccc1)C(=O)NCC(CNC(c1cc(C(F)F)[nH]n1)=O)CO c1(CC)ncc(C(=O)NC2CC(C(C)NC(=O)CC3CSCCO3)C2)[nH]1 c1(OCC(=O)N(CC(C)NC(C(n2cc(C)nc2)(C)C)=O)C)ccc(Cl)c(Cl)c1 C1(NC(c2c[nH]c(Br)c2)=O)CN(C(c2cccnc2C(F)(F)F)=O)CC1O Cc1cccc2c(C(N3CCN(C(=O)CC4CCC4)C(CO)C3)=O)cnn12 c1(C(=O)NCC(O)CO)cc(F)c(F)cc1I.C12CCC(CC1)C(=O)NC2 c1(COC)nc(Cl)cc(=NC2CCN(C(C3CCCC3C)=O)CC2CO)[nH]1 c1(OC)ccnc(CC(=O)NCC#CC2CC2)c1OC c1(C(C(=O)NCC(C)(C2CC2)NC(c2cc(Br)co2)=O)=O)ncccc1O Cc1cc(C(=O)NC2COCC2NC(=O)Cc2ccc(C)s2)c(F)cc1N C1(NC(CCCC)=O)CCC2CCN(C(=O)COCc3cc(C)no3)C1C2 N1(C(CN(C)C(c2cccs2)=O)=O)CC2(CCN(C(C3CCCC(=O)O3)=O)C2)C1 C1(OCCC(=O)NCCN(C2CCCC2)C(=O)CC2CC=CCC2)CCCOC1 N1(C(C(=O)OC)C(C)C)C(=O)NCC(c2ccc(F)cc2)C1=O C1(NC(Cn2c(CCC)ncc2)=O)CN(C(=O)CS(=O)(=O)CC)CC1N=[N+]=[N-] N1(C(CCNC(C)=O)=O)C2CCC1CC(F)(CNC(C1(C(F)F)CCC1)=O)C2 N1(C(c2ccc[n+]([O-])c2)=O)CCC2C(CCN2C(C2CCCCS2(=O)=O)=O)C1 CCS(=O)(=O)c1ccc(CC(=O)N=C2CCN(C)CCN2)cc1 C1(C(N2C(CC(=O)NC3C(C)CN(C)C3)CCCC2)=O)C2CCC(F)(F)C12 C1(C)(CC)CC(NC(=O)C(C)(C)CC2CC2)CN1C(=O)Cc1csc(C)n1 O(NC(=O)C(CC(C)C)NC(=O)C(C)CCC)CCCC=C CCCC(C(=O)N(C(=O)CCc1cccnc1Cl)C)N(C)Cc1nnn(C)n1 C1(CC(=O)N(C)CC2CCN(C(=O)CCc3cn(C)cn3)C2)CCCS(=O)(=O)C1 C12(C(=O)NCC3(OC)CCN(C(c4ccc(Cl)c(N)c4)=O)C3)CCCC1CCC2 C1(C(C(=O)OCC)=O)CCCN1N1CCc2nc(OCC)ccc2C1 C1(C(N2C(C)CCC2C)=O)CC2(CC(NC(=O)Cc3cnn(C)c3)C2)C1 C(=O)(C(CO)NC(c1cc[nH]n1)=O)NCC(CC)N1CCCC1 C=CC(CCC)CC(=O)NCC1(NC(c2ccc(OC(C)C)nc2)=O)CCOC1 C1(NC(c2c(C)nc(CO)s2)=O)CCCN(C(=O)Cc2ccsc2C)C1C c1(OC)c(C(=O)OCCc2ccsc2)cccc1C(=O)O c1(C(=O)NCC(CC(C)C)NC(=O)Cn2ncnn2)ccn2c1CSCC2 c1(C(N2CCC(COC)(NC(=O)C(C)C(C)C)C2)=O)ccncc1N=[N+]=[N-] O(NC(=O)CC=CCNC(C1CCC(C(N)=O)O1)=O)CCCC=C Cc1ccc(C(N2CCCCC2CCCO)C(=O)NCC2CCCO2)cc1F c1(C(N2CC(NC(COCC)=O)C(C(F)(F)F)C2)=O)n[nH]c2c(OC)cccc12 C12(C(N3CCC(CNC(C(CC=C)(C)O)=O)(COC)C3)=O)CC1COC21CCC1 O=C(CC1CCOc2ccccc21)NCC1(NC(C2CCS2(=O)=O)=O)CCCC1 N1(C(C=C(C)c2ccco2)=O)CCN(C(C23CCC2C3)=O)CC1C(C)(C)C c1(CCC(N2CC(NC(C(C)(C3CCOCC3)OC)=O)C2)=O)cc(C)nc(C)c1 N#CC1=C(C(=O)NCC2(CNC(=O)C(N)=O)CCOCC2)CCC1 C1(NC(CCCOCC=C)=O)C2CCC1N(C(=O)C=Cc1ccc(C(N)=O)o1)C2 Cc1ncc(C(=O)NC2(CCO)CN(C(=O)Cn3cnc(Br)c3)C2)s1 C(=O)(CC(C(F)(F)F)c1cccc(F)c1)NC(CNC(c1c(C)scn1)=O)CO CCCCCC(CC)C(=O)NCC=CC(=O)NCCC(=O)N1CCCC1 C(C1CN(C(C2CCCC2OCC)=O)CC1C(=O)N(C1CCC1)C1CC1)=CC c1(C(N2CCN(C)C(CNC(C3(C(F)F)CC3)=O)C2)=O)cnn2ccccc12 c1(-c2nc(CCCOC)nn2Cc2cnc3[nH]ccc3n2)ccc(S(C)=O)cc1 CCC(C#N)C(=O)NCc1ccc(C(N2CC(NC(=O)N(C)C)C2)=O)cc1 N12CC3CC3(C1)CN(CO)C(=O)C(C)(C)NC(C)C2=O.C(C)(C)(C)OC(C)=O N1(C(C(CC2CCC2)NC(Cc2ccn(C)n2)=O)=O)CCCC(CO)CC1 CC(C)C(F)(CNC(C1(C)CNC(=O)C1)=O)C(=O)N1CC2CCC2C1 C(C(=O)NNC(=O)C1CCOC1C(C)(C)C)C1(OCC)CCCC1 c1(N2CCCC3(N(C)CCC3)C2)cc2ccc(Br)cc2c(Cl)n1 c1(NC(C(CNC(=O)CSc2cn[nH]c2)O)=O)cccc2[nH]ccc12 C(C(C(=O)N1CCC(c2nc[nH]n2)C1)NC(=O)CCc1cnco1)N(C)C C1(NC(COCCC(C)C)=O)C2CCCN(C(=O)CC3OCCC3C)C2C1(C)C CC1(C(=O)NCC(C)(C2CC2)NC(C2CCS(=O)(=O)CC2)=O)CC2CCC1C2 c1(N(CC(CN(C(=O)CC2CC(=O)NC(=O)C2)C)O)C)ncc2ccccc2n1 Nc1cc(C(=O)NC2CCN(C(C3CCCOC3)=O)C2)ncc1Cl c1(NC(=O)NC(C#CCC)(C)C)nc2ccc(N)cc2s1 c1(C)ccc(Br)cc1.C1(C)(C(C)C)CC1NC(N1CC(O)C1)=O c1(NC(CCCNC)C)nc(C(C)C)ncc1Br.CS Cn1cc(C(N)=O)c(NC(=O)CCC2(C)CN(C(C3CC3C3CC3)=O)C2)n1 C1(NC(c2c(OC)csc2)=O)CN(C(c2cccc(F)c2N)=O)CC1(C)C N1(C(c2scnc2Br)C(=O)NC2CCOC2)CCCCC1CF CC1(CNC(=O)C=CCn2cncn2)CCCN(C(C2OCC3CCCC23)=O)C1 C1(C(=O)NCC2(C(=O)NC3(C(=O)NC)CC3)CC2)CC1(F)F C(C(C)(C)C(=O)N1CCCC(CN(C(=O)CC2(OC)CC2)C)C1)OC N1(C(CC(CC)OC)=O)CCC2(CCC(C(=O)NCCC3CCCC34CC4)O2)CC1 c1(CC)nc(C(N2CC(CCCCNC(c3ncoc3C3CCC3)=O)C2)=O)co1 c1(OC)ccc(CO)cc1C(=O)NC1CC(NC(=O)CC2CCCC2(F)F)C1 C(=O)(CCCC(F)F)NCC1OCCN(C(C2(CC)CCCC2)=O)C1 c1(C(N2CCCCC2(C)P(C)(C)=O)C(=O)NC(C)(C)C)ccc2cnccc2c1 CCC(CNC(=O)C(C)CN(C)C(C1CNC(=O)N1)=O)(CC)CO c1(C(N(C(CNC(Cn2c(C)ccn2)=O)C2CC2)C)=O)coc2c1C(O)CCC2 N1(CCC(C)C(F)F)C(=O)CCN(C2CC(C)(C)Oc3cc(F)cc(F)c32)C1=O C1(C(N2CC(n3cc(C4C5COCC45)nn3)C2)=O)(OCC)CC2(CC(F)C2)C1 CCC(C#N)C(=O)NCC(C)N(C(=O)CCCc1cnn[nH]1)C Cc1cc(C(N2CCCC(C(C)NC(c3ccc(Cl)s3)=O)C2)=O)cc(C)c1C#N N1(C(C2N(C(C)=O)CC(O)C2)=O)CCC(NC(c2ccnnc2)=O)C12CCC2 C(=O)(C(C)(C)C(F)F)NC1CC(F)(CNC(C(C(C)C)SCC)=O)C1 c1(C(N(CC(CNC(C2(COC)CC=CCC2)=O)(C)C)C)=O)cc(C)cc(C)c1 C(=O)(CC(O)C(C)CC)N1CCN(CC(=O)NC2CON(CC)C2=O)CC1 C(=O)(CC(CCCC(C)C)NC(=O)C(c1ccccc1CC)O)OCC C(CCCCC1CC1)(C(=O)NCC(=O)OC)N(CC=C)Cc1cccs1 c1(C(C(=O)NC23CC(NC(C4CC(C#C)(O)C4)=O)(C2)C3)OC)cc(Cl)cc(Cl)c1 CCCC(CNC(=O)CC1CC(NC(=O)CC2CCOC2)C1)CCO CC(C)(C)CCCC(=O)NC(CC(=O)N1CCC(n2ccnn2)C1)C(F)(F)F C1(NC(c2c(C)[nH]cc2)=O)CCC2CN(C(C3CC4(C3)CC4(F)F)=O)CCC2C1 C(=O)(C(C#N)C(C)(C)C)NCCCC(C)(C)NC(=O)C(Cc1ccsc1)NC=O CC(C)C(CCc1ccccc1)C(=O)NC(CNC(=O)CNS(N)(=O)=O)C1CC1 C(=O)(C1COc2ccc(Cl)cc21)N1C(C)CC(NC(c2cnoc2)=O)CC1 N1(C(C)=O)CCOCC1CCNC(=O)COC1CN(C(=O)CC(C)(C)C)C1 CCC(CC(=O)N1CC(F)(F)CC1C(C)NC(c1cnn(C)c1)=O)C(F)F N1(C(CN(CCOC)C2CC2)=O)CC=CC(NC(=O)Cc2ccncc2Cl)C1 c1(C(=O)NCC(N2CCC(N(C(CCCOC(C)C)=O)C)C2)=O)ccccc1F CC(C(=O)N(C1CCCN(C(c2ccc(CS(C)(=O)=O)cc2)=O)C1)C)S(N)(=O)=O C(c1ccc(OC)c(O)c1)=CC(=O)NC1C(CC)NC1 N1(C(c2n(CC=C)ccc2)=O)CC2(CCC(CNC(C3CCC4CC34)=O)O2)C1 c12ccc(c(F)c1)C(=O)N1CCCC(O)(C1)CNC2=O.S(=O)(=O)(C1CC1)N.CCN N1(C(c2scc(C#N)c2)=O)CC2CCC1CN2C(C1C2CCCC12)=O N1(C(CCOC)=O)CC(C(=O)NCCc2c(C)noc2C)C(C2CC2)C1 C(=O)(C1=Cc2cc(Br)ccc2OC1)NCCC1N(C(C(C)O)=O)CCSC1 n1(CC(N2C(C)CC(CNC(C(C)=C3CC3)=O)C2)=O)nc2n(c1=O)CCCC2 c1(CN2CC(O)(CNC(c3cccc(COC)c3)=O)C2)ccc(F)c(C#N)c1 Cc1cnc(NC(C2CCCN(C(=O)OC(C)(C)C)C2)C)c([N+](=O)[O-])c1 CC(C)CCC=CC(N1CCC(NC(C2(Cl)CC2(F)F)=O)C1)=O N1(C(c2ccc(C)nc2C)=O)CC(NC(C2CC(C)(O)C2)=O)C(S(C)(=O)=O)C1 C1(CNC(C2(F)CC2)=O)COC2(COCCN(C(C3(F)CCCC=C3F)=O)C2)C1 c12cc(S(C)(=O)=O)ccc1CNC2=O.C1(CC)CCN1C(=O)C(O)C1CCC1 C(=O)(CCCC(C)(c1nnnn1C1CCC1)NC(c1ccc(Br)cc1F)C)OC CCCCC(C)C(=O)NC1C=CCN(C(=O)CSc2nnnn2CC(F)(F)F)C1 C(CC(C)(C)C)NC(N(C1CC(F)(F)C1)CCC#C)=O [N-]=[N+]=NCCCC(=O)N1CC2CC(C1)N2C(=O)C(F)C1CCOC1 c1(C(=O)NCC(C(=O)NC(C)C(C)(C)O)C)ccn(C)c(=O)c1 N1(C(c2cccc(SCC)c2)=O)CCC2(CCC2)C(NC(C2CC2CF)=O)C1 c1(C(C2(OC)CCN(C(C(=O)OCC=C)=O)C2)OC)ccc(C(F)F)c(Cl)c1 Cc1ccnc(C(=O)NCCOCCCNC(=O)CC2CCCCCC2)c1 c1(OC)ccc(C=CCNC(=O)Nc2nc(Cl)cc(=O)n2C)cc1OC C(CC(=O)NC1(CNC(c2oc(C)cc2C)=O)CC1)(C1=CCCC1)OCC N1(C(C(CO)N(C)C)=O)CC(CNC(C2(C)SCCCS2)=O)C2(CC2)C1 C1(C(=O)NC(c2cccc(OC)c2)C)CCCN(Cc2ccc(F)c(I)c2)CC1 C1(C(N2C(C(=O)Nc3cnn(CCF)c3)C=CC2)=O)CCC2(CC1)CC2 C1(C(C#C)C)CCN(C(C2CCN(C(=O)CN(C)C)C2)=O)CC1 c1(CC(=O)NCC(C)CNC(c2ccccc2CO)=O)cc(Cl)ccc1Cl N1(C(CC2(CC)CCC2)=O)CCC(O)(CNC(c2ccccc2OC(F)F)=O)C1 N#CC1(C(N2CCC(C3CCCN3c3ncccn3)C2)=O)CC2CCC1CC2 Cc1ccc(C(N2C3CN(C(=O)C(C)(C)c4ccccc4)CC23)=O)cc1Cl Cc1cc2cccc(C(=O)NC3CC(C(N4CCN5C(=O)OCC5C4)=O)C3)c2[nH]1 C(C(C)(C)C1=CCCC1)N.C12(C(=O)OC)CCC(NC(=O)CCCC3CC3C)(CC1)C2 N1(C(C(C)Oc2cccc(C)c2)=O)CCC(NC(=O)C=CCO)C12CC2 N(C(=NCCF)NCC1CCC1Cc1ccccc1)C(C1(O)CCCOC1)=O c1(C(N2CC(O)(CNC(CC(C)O)=O)C2)=O)ccc(NCCO)cc1 N1(C(CSCC)=O)CCC(NC(c2cc(Br)co2)=O)C(CC)C1 N1(C(c2ccc(C3CC3)s2)=O)CC(C2CN(C(c3ncc4[nH]ncc4n3)=O)C2)C1 C12(CC(=O)NCC(C)(C)C#N)CCC1CN(C(c1cc(C(N)=O)[nH]n1)=O)C2 C1(C)(NC(C(CC)N(C(=O)CC2NC(=O)NC2=O)C)=O)CCC(C)C1 C(=O)(C(CC1CC1)NC(=O)CN1CC2CC2C1)NC(c1nccn1C)CC c1(CC)cccc(C(=O)NC2CC(NC(C3CCC34CCC4)=O)C(O)C2)c1O n1(CCC(=O)NC2(CC=C)CN(C(=O)CO)C2)cnc([N+](=O)[O-])c1 c1(C(=O)NC2CN(C(COCCC#C)=O)CC2SC)cc2cc(F)ccc2o1 CCCC(C(=O)NCC1(C(N)=O)CN(C(=O)CC2CCC2)C1)n1ccc(SC)n1 N1(C(c2c(N)cc(F)cc2)=O)CC2(COC(CNC(=O)CCOC3CC3)C2)C1 CN1CCOC(CNC(C2CC(O)CN2C(=O)C(O)C2CCC2)=O)C1 C1(OC)CC2(CCC(C(=O)NC3CCC(CCNC(=O)C(C)=C4CC4)C3)CC2)C1 c1(OC)cc(C(=O)NCC(c2ccccc2)N(C)C(C2CC2C)=O)cc(Cl)c1 CC#CCC(C(=O)NCCC1CC1C)NC(=O)CCC(C)CC Cc1c(-c2nc(Cc3ccc(Br)cc3)nn2CC(N)=O)cnc2ccnn12 CCCC(C(=O)NC1(CCNC(c2cc(CCO)on2)=O)CCC1)NC(C)=O C1(NC(C(=O)Nc2ccc(C(=O)NC)cc2)C)CCc2cnn(C(C)C)c2C1 N1(C(C(CC#C)C2CC2)=O)CCOCCC1C(=O)NC(C)Cc1cccs1 CC(CF)CC(=O)N(C)CCN(C)C(c1nc(C(C)(F)F)cs1)=O Cc1nc(O)nc(C)c1CC(=O)NCC(CNC(C1(Cl)CCC1)=O)CO c1(N2C(C(=O)Nc3ncc(Cl)cc3O)CCC2)ncnc2sccc12 C1(C(N(C)CC2(NC(c3cnn(C(C)C)c3N)=O)CC2)=O)CCCC1S(C)(=O)=O N1(C(CCOC)=O)CCCC(CCNC(c2cc(SC)oc2C)=O)CC1 C(C(=O)N(C)OCCCC)(C1C=CCC1)NC(C=CC)=O N1(C(C(CC(=C)Cl)NC(=O)C(C(C)C)NC(C)=O)=O)CC2(CCC(=O)O2)C1 CN1CCC(C(=O)NCCC2(C)CCN(C(c3ccc[n+]([O-])c3)=O)C2)CC1=O CCCC(C)(C)C(=O)NCC1CN(C(=O)C(CCOC)OC)CCCO1 N1(C(CC(CC2CC2)NC(c2cc(C)nn2C)=O)=O)CC(=O)N(C)CC1C C(C(N=[N+]=[N-])C(=O)NC1CCC(C(N2CC(CC(C)C)C2)=O)C1)OCC C1(NC(=O)NC2CCC(CC#N)C2)CC2CC1CC2F C1(CC)CN(C(=O)CN2CC(OC)C2)CCN1C(C12CC(OC)C1C2)=O C(C)(C)(C(C)CC(=O)NC1CC=CCC1)NC(C1CC(C#C)(O)C1)=O c1(C(N2C(CNC(c3cncc(N)n3)=O)CC(F)C2)=O)cc(F)c(F)cc1F C(C)(C(CC(=O)NC12CC(F)(C1)C2)NC(c1cc(N)cc(F)c1)=O)OC C(CCCCCNC(C1CC2CC1C2)=O)N(C)C(C1CC1F)=O C(=O)(CC(C(F)(F)F)OC)NCC1N(C(C=CCC)=O)C2CCC1C2 c1(CCCNC(=O)C(N2CCN(c3cccc(Cl)n3)CC2)=O)ccc(O)cc1 C1(CNC(c2c(C(=O)OC)scc2)=O)C2CN(C(C3CC4(CCC4)C3)=O)CC12 c1(C(=O)NCC(CO)NC(C(COC)C)=O)cccc(N2CCCC2=O)c1 c1(CCC(=O)NC(C2CN(C(CCC#C)=O)C2)C)ccc(F)c(F)c1 C1(NC(COC(CC)(C)C)=O)CCN(C(C23CCC2CC3)=O)C(C)C1 c1(C(N2CC(NC(C3CC(C)(C)C3)=O)C3C2C3)=O)cnn2cc(Br)cnc12 S(=O)(=O)(c1ccc([N+](=O)[O-])c(Cl)c1)NC1C(C(=O)Nc2cncs2)C1 CS(C)(=O)=NC(=O)c1cc(C2OCCO2)on1 N1(C(C(n2cc(Cl)cn2)C)=O)CCCCC(CNC(c2cncnc2)=O)CC1 C1(NC(C2CCC(C)C2)=O)CC1C1CCCN(C(c2ccc3scnc3c2)=O)C1 N1(C(c2c(C(C)C)cco2)=O)CCSCC1C(=O)NCCc1cnnn1C N(C(=NCCC1CCC(=O)N1)NCc1c(Br)nnn1C)C(C)C1CC1 N1(C(C=CC(C)(C)SC)=O)CCC(N=[N+]=[N-])(C(=O)NCC(CO)C2CC2)C1 c1(CC(=O)NCC(C)(C)NC(c2cc(F)cc(N)c2F)=O)ccn2cncc2c1 c1(C(=O)OC)ccc(C(C)NC(C)Cc2cccnc2)nc1 N1(C(c2cc(COC)sc2)=O)CCN(C(=O)CCn2ccnn2)CC1COC c1(C(c2n(CCC)nnn2)Nc2ccc(C)nc2)ccc(C(C)CC)cc1 Cc1ncn2ccc(C(=O)NCC3(CCNC(=O)C=Cc4cccs4)CC3)cc12 Cc1cc(C(=O)N(CCCOCCNC(c2ccn(C)c2)=O)C)c2nccn2c1 N1(C(C(c2ccc(CC)s2)=O)=O)C2CCC1C(C)C(NC(=O)C(C)(O)C(C)C)C2 C1(O)(CCNC(C(C)(C)C2CCCC2)=O)CCN(C(C2C=CCCC2)=O)C1 C(c1ccccc1)=C(CC)C(=O)OC(C)C(=O)C1CCC1 c1(NC(C2C(C(=O)Nc3c(C#N)cno3)C2)=O)ccc(F)c(F)c1O c1(C(=O)NCCOCCO)cccc(F)c1CNC(=O)CCc1ccc(F)nc1 C1(C)(CNC(C(CC)(C)CC)=O)CC(F)(F)CN1C(=O)Cc1ccc(C)c(F)c1 c1(C(=O)NCCC(C)(C)NC(CSCC#C)=O)cc(C)cc(Br)c1F c1(N2CCC(C)(CN(C)C)C2)ccc(S(=O)(=O)NCc2c[nH]ccc2=N)c(Cl)c1 CN1C(=O)NC(C2CCN(CCC(=O)Nc3ccc(I)cc3)CC2)C1=O C1(CC(=O)NC2(CNCc3ccc(CO)cc3)COC2)CC2CCC1C2 CC1CCCc2nc(C(N3CCOC(CCNC(=O)C(C)(C)C#N)C3)=O)cn21 c1(C(=O)NC(CN(CCCCC)CCCNC(=O)OC(C)(C)C)C)cnc(C)[nH]1 CC1CCN(C(C2CC(=O)N2)=O)CC1CNC(=O)C(c1ccc(F)cc1)F C(C(C)(CC(C)C)NCCC(=O)OC(C)(C)C)NC(COCCCCOC)=O c1(OC)nc(N2CC(CNC(=O)Cc3cn(C(C)C)nn3)CC2C)nc(C)c1F C(=O)(CCC(C)(C)F)N1CC(C)C(CCNC(c2ncccc2C(C)(C)C)=O)C1 c1(N2CC(C)C2)ccc(S(=O)(=O)NC2CCN(c3nncs3)CC2)c(Br)c1 C(c1nc2ccccc2o1)=CC(=O)NC(C1CCN(C(=O)C2=CCCC2)CC1)C c1(C(=O)NC2(CO)CCN(C(=O)CSc3n[nH]c(O)n3)C2)cnn2cccnc12 CC1(CNC(C2(C)CC2(F)F)=O)CN(C(=O)COc2ccc(F)cc2Cl)CCO1 Cc1ccc2c(c1)CC(NCC1CCCCN1CC(=O)NC1CCS(=O)(=O)C1)O2 C#CC(CNC(=O)C(C)N(C(c1scnc1C)=O)C1CC1)CC(C)(C)C c1(NC(C(CNC(c2ccc(CC)[nH]2)=O)O)=O)ccnc(OC)c1 N1(C(c2c(CC)nccc2)=O)CCC2CC2(C(=O)NC2(C)CCSCC2)CC1 C12(NC(c3[nH]cc(CC)c3)=O)CCCCC1CN(C(c1nocc1Cl)=O)C2 N1(Cc2nc(C)cc(C)n2)CC=C(CCNC(c2cc(C3CC3)n(C)n2)=O)CC1 c1(C(=O)NCC(C)CNC(=O)CCCS(C)(=O)=O)cccc2cnnc(O)c12 c1(C(=O)NCCCC2(NC(CC3(C)CC3)=O)CC2)cc2n(n1)CCCO2 C1(CNC(C=CC(C)(C)C)=O)CCCCN1C(c1ccc(-n2ccnn2)cc1)=O c1(NC(CC2(C)CN(Cc3c(OC)ncnc3OC)C2)=O)cccc2nc[nH]c12 C12(CNC(C3C(C)=C3)=O)CCCC1N(c1ncnc3ccsc13)CCC2 C12=NC(=NCC(C)CNC1=O)C=CN2.C1(CC(=O)N(CC)CC)CCCOCC1 c1(C(=O)NC2(CO)CCCN(C(C3CC(N=[N+]=[N-])C3)=O)C2)nc2c(s1)COCC2 C(C(=O)NCc1ccc(C)nc1)(C(C)CC)NC(c1ccc(NC)cc1)=O c1(N2CCC(CCCC)C2)nc(N2CCC(CC(F)(F)F)C2)cc(C)n1 C=CC(C)(CC)C(=O)NCC(C)(CO)NC(=O)COc1ccsn1 CC1CCCC1N=c1nc(N(CCCN2CCCC2)C)c2sccc2[nH]1 c1(C(=O)NC(c2cccc(C)c2)CNC(C(CC)F)=O)ccc(C2CC2)nc1O c1(OC)ccc(C(C)Nc2ccc(NC(C3COC(=O)N3)=O)cn2)cc1 C1(F)(CNC(C(C)OCC2CC2)=O)CCN(C(=O)CCc2ccccc2Cl)C1 CCCC(O)CC(=O)NC1CCCC1NC(c1cn(CCC2CC2)nn1)=O C1(SC)COCC1NC(=O)CCCN(C(=O)C(C)OCC1CC1)C C1(NC(c2cc[nH]c2C2CCCC2)=O)CC2CN(C(=O)C(F)=CC3CC3)CC12 CC1CC(NC(C2OCCC2NC(=O)CC2CSC2)=O)c2nccn21 C#CC1(C(=O)Nc2cccc(OC)c2C)CCN(C(=O)CC2CC(CC)=NO2)C1 CCCC(CC)C(=O)N(CCCOCCN(C)C(c1cnc(C(F)F)s1)=O)C N1(C(C2N(C)CCC2)=O)CCC2(CC1)OCCC2NC(C1(CO)CC1)=O N1(C(c2c(OC)ccc(C)n2)=O)CC2CS(=O)(=O)CC2(NC(=O)C(F)F)C1 N1(Cc2cn(C(c3ccc(C#N)cc3)CF)nn2)CCOC2(CCOC2)C1 C1(COC)(NC(c2cc(CO)[nH]n2)=O)CN(C(=O)CCc2ccc(Cl)s2)C1 Cc1cc(C(F)F)oc1C(=O)NCC(CO)NC(=O)Cc1cnccn1 c1(CNC(C2(C(N)=O)CC2)=O)ccc2c(c1)CCN(C(C1CC3CCC3C1)=O)C2 c1(OC)ncc(CN2CCC(NC(=O)Cc3ccc(Cl)cn3)C(F)C2)cc1C N1(CCC(N2CC(CC)C(N)CC2)=O)C(=O)Cc2ccccc2C1=O N1(C(C(C(C)C)CNC(=O)CC(C)n2ccnc2)=O)CC2(C)CCC2(C)C1 N1(C(CN=S(C)(C)=O)=O)CCC2(CCOC2)C(CNC(=O)C2=CCCOCC2)C1 C1(O)(CNC(CC(C)N(C)C)=O)CCN(C(=O)Cc2cc[nH]c2)C1 O=C(NOCCO)C1c2c[nH]nc2CN1C(=O)C1=CC2C=CC1C2 CC(C)C(C#N)C(=O)N(C(C)CCNC(c1cccc(F)c1Br)=O)C C1(O)(CN(C(=O)Cn2cc(Cl)cn2)C)CCN(C(=O)Cn2cnnc2)C1 CC(C)CC(CNC(C12CCC(C)(C1)OC2)=O)C(=O)NC1CC12CCC1(CC1)CC2 CC1COC(CO)CN1C(c1c[nH]nc1CNC(c1ncncc1Cl)=O)=O C1(COc2ccc(Cl)cc2)CC2CCCC2O1.c12cccc(c1)C(=O)NC2 n1(CC(=O)N(CC(CN(C(CCCc2ccc(C)s2)=O)C)O)C)cc(Cl)c(C)n1 c1(C(=O)NC2CCCC2CNC(C2(F)CCOC2)=O)ccncc1C(F)F c1(C2CCN(C(=O)NCC3(CSC)CC3)C2)nc2ccccc2o1 C(=O)(CC1=CCCCC1)N1CCC2C(NC(c3c(C)c(F)ccc3)=O)C2C1 c1(C(=O)NCC2C(NC(C(CSC)C)=O)CC2)nc(C2CC2)ncc1Cl CC1(C)C2CCC1(C(=O)NCCNC(C1CCc3ncnn3C1)=O)CC2 C(C(C(=O)N(C)CCNC(C1CCCN1CCC(C)C)=O)OC)OC c1(CN(C(=O)CC2C(C)(C)C2(C)C)C)nnc2n1CCCC2C(F)(F)F c1(OC)nccc(C(=O)N(C2(CC(=O)NCCCN3CCNC3=O)CC2)C)n1 c1(C(N(CC(C)O)CCNC(C(CC)F)=O)=O)ccnc2[nH]c(CC3CC3)nc12 N1(C(C2(CC)CC2(F)F)=O)CCN(C(=O)Cc2cc(C(C)C)no2)CC1C c1(C(=O)NC2CC3(C(NC(C(CC=CC)C)=O)C3)C2)c(O)nnc2c1COCC2 n1(CC)cc(Cl)cc1C(=O)N(C)CCN(C(c1sc(OC)nc1Cl)=O)C(C)C C1(C(N(CC(C)(C)NC(=O)CN2CCCCC2)C)=O)CC12CCC1(CC1)CC2 C1(CCSC(F)(F)F)CC2CN(CC(=O)NC(CCCCC)=O)CCN2C1=O C(=O)(C(C)(C)C(F)(F)F)N1C(CNC(c2c(O)ccc(CC)c2)=O)CC1 C1(C(C)NC(C(N2CCOC2=O)C)=O)CCCN1C(=O)CCn1cnnn1 N1(C(CCC2C(=O)NC(=O)N2)=O)CC2CCC1CN2C(c1nccc(Cl)c1O)=O N(C1CCCNc2ccccc21)C(=O)NCCCN1CCOCC1 c1(C(=O)NCC2(F)CC(NC(=O)C=CCO)C2)ncnc2ccsc12 CCC(CNC(C1(CCOC)CCC1)=O)(CC)NC(=O)C(c1ccc(C)cc1)C Cn1c(C(=O)NCC(F)CNC(=O)C(C2CCCCC2)F)cc2ccc(O)cc12 N1(C(c2ccc3c(n2)OCCO3)=O)CCC2(CCN(C(C3CC(O)C3)=O)CC2)C1 N(C)(S(=O)(=O)NC(c1cccc(Cl)c1)C)C(C1CCCC1)C c1(NC)ccccc1C(=O)NC1CCC1C(=O)NC1CCC(C(N)=O)C1 c1(N2CC(CC(C)NC(C34CCCCC3C4(F)F)=O)C2)cc(C)c(C#N)cn1 c1(C(=O)NC(C(=O)OCC)C2CC2)ccoc1CNC(c1cncn1C)=O c1(OC)cc(C(=O)CCC(=O)NCCNC(c2ccccc2SC)=O)ccn1 c1(C(N2CCC(S(C)(=N)=O)CC2)C(=O)NCC=C)cc2ccnc(Cl)c2s1 c1(C(=O)NC(CCSC)Cc2cccnc2)ccc(Br)c2c1OCCC2 N1(C(c2nnc(C)s2)=O)CCC2(CC1)CCN(CCC1CC1)C2 Cc1cc(C(C)(C)C(=O)NCCNC(=O)CC(O)c2cc(C)cs2)cs1 CC1Cc2ccc(F)cc2C1NC(=O)Cc1c[nH]c2ccccc12 c1(C(N2C3(CNC(C4CCCC4)=O)CCCC3CC2)=O)cc2n(n1)CCNC2=O c1(C(C)NC(C(CC)O)=O)ccc(CNC(=O)CNC(=O)C2CC2)cc1 c1(C(=O)NCCCCN(C(=O)CCS(C)=O)C)cn2c(n1)COCC2 C12(C(N3C(C)CCC(CNC(C(C)OCC=C)=O)C3)=O)C3C4C1C1C2C3C41C c1(NC(CCCC)c2nnnn2CC2CCOC2)ccc(SC(F)F)cc1 C(=O)(C1=CCCOCC1)N1CCC(N(C(Cc2c(COC)cccc2)=O)C)C1 C1(CCNC(CSCCC)=O)C(C)CCCN1C(c1scnc1C)=O Cc1nccc(Cl)c1C(N1CC2C(NC(c3ccc[nH]3)=O)C2C1)=O C1(C(=O)NCc2snc(CC)n2)CCC2(CC2)N1C(C1CN(C(C)=O)C1)=O C1(C(N(CCCCO)CC)=O)CC(=O)CN1C(=O)C=C(C)C C1(NC(c2cc(CC)[nH]n2)=O)CC2CC(NC(c3cscc3C(F)(F)F)=O)C1C2 c1(N(C)C)ccc(S(=O)(=O)NCC(N2CCC3NCCC23)=O)cc1[N+](=O)[O-] C(=O)(CCC(F)(F)F)NC(C(=O)NCC(CO)N(C)C)CCF Cc1cccc(Br)c1C(C(=O)N(C)CCC1CCCO1)NC(C1CC1Cl)=O c1(C(N2CCC(C=C)(C(=O)NOCCN(C)C)C2)=O)cccc2cc[nH]c12 C#CC1(C(=O)NCCCc2cnn[nH]2)CCN(C(C2CC(O)CN2C)=O)C1 N1(C(C=C(CC)C)=O)C2CCC1C(C)C(NC(c1nc(C(F)(F)F)cn1C)=O)C2 CCC(CC)(CC)C(=O)NCC(c1ccccc1)NC(c1cnn(C)c1N)=O C1(CC)CCCN(C(c2cnn(C)c2Cl)=O)C1C(=O)NC1CCCC1O Cc1cc(C)cc(S(=O)(=O)N2CCCC(C)(C(N3CC3C)=O)C2)c1 C1(C2CCN(C(=O)Cc3cccc(O)c3)C2)(NC(CC2C(C)=NOC2=O)=O)CC1 C(CCN=c1[nH]c2ccc(O)cc2s1)NC(c1cn(C)c(=O)n(C)c1=O)=O c1(CN2C(C(=O)OC)CC(NC(c3ccnc(C)c3)=O)C2)ccc(NC)cc1Cl c1(CC(=O)NCC(C)CN(C(=O)C(F)CC)C)nc([N+](=O)[O-])n[nH]1 Cc1cc(C(=O)NC(CNC(=O)C=Cc2nccs2)C2CC2)cc(C)n1 C1(CC)CCC(C(N2CCN(CCN(C)CC3C4CC5C(C4)C35)CC2)=O)CC1 C1(F)(C(N(CC(CC)NC(c2cnc(O)cc2OC)=O)C)=O)CCCN(C)C1 N1(C(C2N(C(c3ccc(C4CC4)o3)=O)CC(=O)NC2)=O)CC2CCC1C(O)C2O C=C(CNC(=O)C(OC)OC)CCNC(c1[nH]nnc1C(F)F)=O Cn1nc2c(c1C(N1CCCC(F)C1)=O)CN(C(=O)C1CC1)CC2 N1(C(CN(C(=O)OCC)C)=O)CCCC(O)CC1C(=O)N(C)CCc1cccs1 C1(C(N(CCCC(=O)NCc2ccc(C#N)s2)C)=O)CC(F)(F)CO1 c1(C(N2C(C(=O)Nc3ccccn3)CC3CC32)=O)c(F)cncc1Br c1(NC2(CNC(C(CC)N(C)C)=O)CC2)cc(C(C)C)nc(COC)n1 c1(C(=O)NC(CNC(c2ncccc2F)=O)C2CC2)ccc2c(c1)CC2 C1(NC(COC2(C)CCCC2)=O)CN(C(C2CCCOC2)=O)Cc2ccnn2C1 c1(NCC(C)CCO)nccc(=NCc2nnc(Br)n2C)[nH]1 C(C(CC(F)(F)F)NC(C1CC1C1CCC1)=O)NC(=O)C=CCN1CCCC1 c1(C(N2CCC(NC(c3c(C)noc3N)=O)C(F)C2)=O)cccc2occc12 CC(C)CC(CNC(=O)COCCOCCO)NC(c1n[nH]cc1F)=O N1(C(CC=C(C)C)=O)CC(CNC(c2cnn(CC(F)F)c2)=O)C(F)(F)C1 Cc1cnc(C(N2CCN(C)CC2C(N2CCOC(C)(C(C)C)C2)=O)=O)cc1C Cn1ccc(CC(N2CCC2C(=O)N(CC(N2CCOCC2)=O)CCO)=O)n1 Cc1cc(F)cc(C)c1C(N1CC(NS(=O)(=O)CC#N)C(C#N)C1)=O C=C(C)CCCC(=O)NC1CC2(C1)CC(C(N1CCC(C)CC1C(=O)OC)=O)C2 C1(N(C(Cc2nc(C)sc2)=O)C)CN(C(=O)CC2(N3CCCC3)CC2)CC1O CCC(C)(COC)C(=O)NC1CN(C(=O)CCNC(c2cccs2)=O)CC12CC2 c1(C(=O)NCC(C)(CO)NC(C(CCCOC)C)=O)ccnc2c1CCO2 c1(C(N2CCC(N(C)C(C34COCC3C4)=O)C2)=O)cc(C2CC2)ccn1 N1(C(C(COC)NC(C)=O)=O)CCC2CCCC(C1)N2C(=O)Cc1cncn1C C1(NC(C2CCCCCC2)C(=O)O)CN2CCC1c1ccccc12 CCCC(C(=O)NCC1(O)CN(C(=O)CSC(F)(F)F)C1)OC C#CCC(C)(C(=O)N(C(C(N)=O)C1CC1)C)NC(C1CCC(=O)NC1)=O c1(CN=C(NC2C(C)NC(=O)CC2)NCc2ccco2)cnn2ccccc12 C1(NC(c2c(C)c(O)ccc2)=O)CCN(Cc2cccc3[nH]ncc23)CC1(C)C C1(CC(N)=O)CCN(C(=O)COCCNC(c2cnc(C(F)(F)F)cn2)=O)CC1 C1(CC=C)(NC(c2cnncc2NC)=O)CCN(C(=O)C(F)C(C)C)C1 N1(C(CC)=O)CCC(NC(c2cc(=N)[nH]cc2Br)=O)C(F)(F)CC1 N1(CC(C)NC(C2CC3CCC2O3)=O)CCN(C(C2(C(C)(F)F)CCC2)=O)CC1 C1(CC(=O)NCC(C(C)C)NC(c2ncsc2C2CC2)=O)CCC(C)(C)CO1 CCCC(O)C(=O)NC1CCN(Cc2nccn2CC)C1 c1(C(=O)NC2C(NC(C3(COC)CCCO3)=O)CCC2)onc(C)c1C CS(=O)(=O)c1ccc(NC2(CNC(=O)C3=CCS(=O)(=O)C3)CCCC2)nc1 c1(C(=O)NCC(C)NC(c2cc(CCC)c(C)s2)=O)n[nH]c(CC)c1[N+](=O)[O-] N1(S(CCN2CCN(C)CC2)(=O)=O)CCN(C(=O)OC(C)(C)C)CC12CCCC2 C1(CNc2nc(C)nc(O)c2)CC2CCC1N(C(C1(CO)CCOCC1)=O)C2 c1(CC(=O)NCCCCC2CN(C(C3CC(C)OC3)=O)C2)ccccc1[N+](=O)[O-] c1(C(=O)NCC2C(NC(C(C)C3CC3)=O)CC2)ccc2c(cnn2C(F)F)c1 C1(NC(C(CCC)C)=O)CN(C(=O)Cn2ncc(Br)c2C)CC12CCC2 c1(C(N2CCC(F)(CNC(CCC=C=C)=O)C2)=O)c(OC)ccnc1OC C(=O)(C1=CC2(CCOC2)C1)N1CC(CCNC(C(c2cn(C)nc2)(F)F)=O)C1 C1(C(=O)NCCC2CCN(C(c3nc(COC)oc3)=O)CC2)CCCC2(CC2)C1 C12CCCN1NC(=O)CONC2=O.Cc1ccc(CCN(C)C(C)C)cc1 N1(C(CN(C)CC)=O)CCCC2CN(C(C3(C4=CCCCCC4)CC3)=O)CC12 C(C(CO)(CO)NC(=O)CC1(C)CC1F)N(C(=O)CNC=O)C C1(C(C)O)CCCN1C(=O)CCN(C(=O)C(F)C1CCOC1)CCO C(CC(=O)N(C1CC2CCC(C1)N2C(=O)C(C)(C)OC(C)=O)C)(C(F)(F)F)OC c1(C(=O)NCC(CC=C)NC(=O)Cn2ccnn2)ccnc(OCCO)c1 c1(OC)cc(C)c(C(=O)NC(C)CN(C)C(C2CCCO2)=O)c(F)c1 N1(C(C(C)CNC(=O)C(F)n2ccnc2)=O)CCCCN(C)CC1 N1(C(C2(C)CC2(F)F)=O)CCC2(CC1)C(NC(c1cc(CO)on1)=O)CS2(=O)=O c1(C(=O)NC(C)CNC(C2CC(=O)NC(=O)N2)=O)ccc2c(C)cc(O)nc2c1 C1(NC(C(C)(C)SC)=O)CC(C)N(C(=O)C(C)OC2CCCCC2)C1 c1(C(N2CCC(NC(CCCC#C)=O)(COC)C2)=O)cc(F)cc(C)c1O C1(NC(CC(CC)C2CC2)=O)C2CC3C(C2)C13C(N1CC(N=[N+]=[N-])C1)=O CC(=O)CCCC(=O)NCC1(O)CCCN(C(=O)CCC(=O)c2ccc[nH]2)C1 CN1CC(NC(=O)CNC(=O)CNC(c2ccc(CO)o2)=O)C2(CC2)C1 C1(CC)C(NC(=O)CCOCC2CC2)CCN1C(C1OCCCO1)=O N1(C(c2c(CC)nns2)=O)CCN(C(c2coc(CS(C)(=O)=O)n2)=O)C(CO)C1 C#CCCC(O)C(=O)NC1(C(=O)NCc2cnn(-c3ccccc3)c2)CCCC1 CC1Cc2cc(F)ccc2N(C(=O)NC2CC(=O)N(C(C)C)C2)C1 C1(C(N2C(C(N(C3(C4CC4)CC3)C)=O)C=CC2)=O)CC2(CCO1)CC2 c1(N2CC3(CN(C(C(CC)NC)=O)C3)C2)ncnc2cc(OC)c(OC)cc12 CC1(CNC(C2(CC3CC3)CC2)=O)CCC(NC(=O)CCc2cc(Cl)cs2)C1 c1(NCCc2ncc(CC)s2)nc(N2CC=CCC2)nc2scnc12 N1(C(CN(C(C)C)C)=O)CC(=O)CC1C(=O)NC1CC(CF)C1 Cc1[nH]nc(C(N2CCN(CC(=O)N(CCCF)C)CC2)=O)c1Cl c1(C(=O)NCCC2N(Cc3cc(C)sc3C)CCC2)cccc(C)c1C C=CCCC(F)(F)C(=O)NCC(C1CCC1)NC(C1(C)CCCNS1(=O)=O)=O c1(C(=O)NC2(c3cn(CC4CC(C)SCC4)nn3)CCC2)cc([N+](=O)[O-])n[nH]1 N1(C(CCc2cc(C)no2)=O)CCC(C)C(CNC(C2(COC(C)C)CC2)=O)C1 c1(C(=O)Nc2cc(F)cnc2Br)cc(-c2c(F)cc(O)cc2F)c2n[nH]cc2c1 O=C1CCC(CC(=O)NCC2CCN(C(C3(F)CC=CCC3)=O)CC2)CN1 c1(C(N(C(C)CNC(C2(c3cccnc3)CC2)=O)C)=O)cc2n(n1)CC(F)C2 N1(C(c2ccc(NC(C)=O)cc2)=O)CCC2(C1)CN(CC(=O)N=c1cco[nH]1)C2 c1(C(C)C)ncncc1C(=O)NCCN(C1CCCC1)C(=O)CC1CC1C c1(C(N2CCC(F)(CNC(COCCC)=O)C2)=O)cnc2c(C)cccc2c1 C1(NC(C(C)(C2CC2)NC(C)=O)=O)CCCCN(C(C2CC(F)C2)=O)C1 C(c1nc2ccccc2[nH]1)=CC(N1CC(CC)N(C(c2cnc[nH]2)=O)CC1)=O Cc1ccc(Cc2nc(C3(C(=O)NC4CCCC4)CC3)nn2-c2ccccc2)cc1 CCCC(C)(O)C(=O)N1CCC(C(=O)N(CC(C)SC)C)O1 O=C1CCCC(C(=O)NC2C=CC(CC(=O)NCc3cnn(CCF)c3)C2)N1 C1(CC(N2C(C#C)CCC2)=O)CN(C(c2cnn(C(F)F)c2)=O)CC12CC2 C1(N(C(C2CCCCO2)=O)CC)CC(=O)N(C(C)C2CC2)C1 CCC(C)(C)CCCC(=O)N(CCNC(=O)CC1OCCO1)Cc1ccccc1 Cc1oc(Br)cc1C(N1CC(F)CC1CNC(c1cnn(C)c1C)=O)=O CCC(=O)CCC(=O)NCC(O)CNC(=O)CC1COCC1(C)C c1(C(=O)NCC2CN(C(C(COC)OC)=O)C3(C2)CCC3)ccc(C#N)c(C)c1 N1(C(C(c2ccoc2)NC(c2c(C)cc(N)cn2)=O)=O)CC(C2=NOC(C)C2)C1 CC(C)C(F)(CNC(=O)CCCC1CCCO1)C(=O)NC(C12CC(CO1)C2)C c1(CCC(=O)NC2(C)CN(C(CC(CC)CC)=O)C2)nc2cnccc2[nH]1 N1(C(C2C(C)CCOC2)=O)CCN(C(c2csnn2)=O)C(c2cccnc2)C1 c1(C(=O)NC2CCCN(Cc3cc(OC)ncc3)C2)ccc([N+](=O)[O-])o1 c1(OC)cc(C(=O)NCC2C(C)CCN2C(=O)CCCC#N)sc1Br C(=O)(C1=CCC(NC(C2CC2(F)Cl)=O)C1)N1C(CC)(CC)CC1 C12(NC(=O)C=CCN3CCOCC3)CCN(C(=O)CC3CCOC3)CC1C2 C1(NC(=O)NCC(c2ccc(F)cc2)Oc2ccc(Cl)cc2)CCCC12CCNC2 c1(C(N2C(C)CCC(CNC(C3(C(=O)OC)CC3)=O)C2)=O)ccc2cnsc2c1 C1(NC(=O)CCC2CC2(F)F)CC12CCN(C(C1(CF)CCC1)=O)CC2 Cc1cc(O)ncc1C(=O)NC(CO)CCCCNC(=O)CN(C1CCC1)C c1(CNC(=O)NC2CC2c2ccccc2OC(F)F)cc(C(F)(F)F)ccc1F c1(NC(c2n(C(C(=O)OC)C)nnn2)CC(C)C)ccccc1CCCO C1(OC)CC(CNC(c2cnc(C(C)C)o2)=O)N(C(c2cccc[n+]2[O-])=O)C1 C1(F)(C(=O)NCCC2(NC(CC3C(C)OCC3)=O)CCCC2)C(C)(C)C1(C)C c1(C(N2C(CNC(CS(=O)(=O)N(C)C)=O)CCCCC2)=O)cccn2nnnc12 c1(OC)cc(C)ccc1C1(CNC(=O)Nc2nccs2)CC1 C(CCN=c1[nH]c2c(c(=NC(C)c3nc(=N)[nH][nH]3)[nH]1)CCC2)SCC Cc1nc(C(C)C)oc1C(=O)NC(C)C(C)(C)NC(c1cnc(=N)[nH]c1)=O c1(C(C)C)ccc(C(CNC(=O)CN2CCCC2)NCc2cc(C#N)no2)cc1 c1(C(=O)NCCC(CC)(CC)NC(CSCCC)=O)ccc(F)c2c1CCC2 c1(C(N(c2ncc(C(=O)OCC)s2)C)=O)cc(C)n(-c2cc(C)on2)c1C C1(NC(C=C)=O)CCN(C(c2ccc(NC)cn2)=O)CCC1c1ccccc1 Cc1cc(CC(N2CCOC(CNC(c3ncnc(C)c3C)=O)C2)=O)cc(C)c1 N1(C(C2C(CCC)C2)=O)CC2(C1)CN(C(c1cnco1)=O)CCO2 c1(C(=O)NC2CN(C(C3C(OC)(OC)CC3)=O)CC(O)C2)ccn2ccnc2c1 Cc1cc(C(N2CCC(C)(CNC(C34CC(O)C3C4)=O)CC2)=O)c(N)cc1F c1(C(=O)NCCC2(O)CCN(C(C(C)OCCC=C)=O)C2)cc(F)cc(Cl)c1 C1(C(=O)NC2C(C)N(C(=O)CCc3cn[nH]c3)CCC2)CC2(CO1)CC(F)(F)C2 CCS(=O)(=O)c1cccc(CC(=O)NC23CC(NC(C4CCCCS4)=O)(C2)C3)c1 c1(CC)cccc(OCCOCC(O)CN2CCOCC2)c1 c1(CN(C(c2nc(CCC(=O)NCCSC)cs2)C(=O)OC)CCC)cnn(C)c1 C(=O)(CN=c1cc[nH]cc1)NC1CC(NC(C=Cc2ncn(C)c2)=O)C1 C(CCC(=O)NC(CN(C)C)C(=O)NCC1COCC1O)OC(C)=O c1(CC(=O)OCCC2CCCC(C(F)(F)F)O2)cccc2cnccc12 N1(C(C2N(C)CCCC2)=O)CCOCC(NC(=O)C=CC2COC(C)(C)O2)C1 Cc1cc(=NCC2(C)CCCCO2)[nH]c(N2CC3CCC2CN3c2ccccc2)n1 c12cnc(c(C)c1)N(S(C)(=O)=O)C1CCN(CC1)C2=O.CCON N1(C(C(C2CCN(C(=O)COCCF)C2)F)=O)CCC=CC1CO N1(C(COCCOCC)=O)CCC(NC(=O)C=Cc2ccncn2)CC1 C12(NC(C3OCCN(C(C(C=C)O)=O)CC3)=O)CC3CC(CC1C3)C2 C1(N(C(C=CC(=O)N(C)C)=O)C)CCN(C(=O)CSc2cnn(C)c2)C1 CN1CCC(C(=O)NCc2n[nH]cc2C(N2CCC(N3CC(O)C3)C2)=O)CC1 C(CNC(c1c(C)nn(CCO)c1C)=O)(C(C)C(C)C)NC(CCOC)=O CCC(C)(C)CC(=O)N1CCCC(N(C(=O)CC2COCC(C)(C)O2)C)C1 C(C(=O)NOCCO)(C1CCCO1)NC(C(CN(C)C)O)=O C(C(C)(O)CC(=O)NC12CC(C1)N(C(=O)C=CC1CCCCC1)C2)OC C(=O)(C1CCCc2cncn21)N1CCC(CN(C)C(c2cc(N)ccc2F)=O)C1 c1(C(=O)NCCCC(C)NC(=O)CC2CCOC2)nc(F)ccc1Cl C(N=c1[nH]c(=NCC(C)CSCC)c2ncccc2[nH]1)c1c(OC)cccc1F N1(C(CNC(=O)NC)=O)CCC2(CC1)CCN(C(c1ccnc(C)c1C)=O)C2 c1(C(=O)NC2C(NC(c3c(SCC#N)cccc3)=O)C2)nnn2c1C(=O)NCC2 c1(CC)cccnc1N1CCC(CCC(=O)NCC(c2cccc(F)c2)C)CC1 Cc1ocnc1C(=O)NCC(C)(C)NC(C12CCCC1C2)=O C1(C(=O)NCC2(O)CC(CO)C2)(NC(=O)CC2(O)CCC2)CC(O)C1 C=CC(O)C(=O)NCC1(CNC(C2CC=CCC2)=O)CC1 c1(C(=O)NCC(CCCC)NC(c2cc(C)nc(O)c2)=O)cc(Cl)nc(Cl)c1 c1(NCCCCNC(C2C3(CC(C)(C)C3)C2)=O)ccc([N+](=O)[O-])cc1S(C)(=O)=O c1(C(N2CCN(Cc3cc(C)c(O)cc3)CC2)=O)c[nH]c2ccc(Br)cc2c1=O c1(C(=O)NCC(C)(O)CNC(C2(C#N)CC3(CC3)C2)=O)ccc(S(N)(=O)=O)cc1 N1(C(c2c(C)ccc(OC)n2)=O)CCC2CN(C(=O)C(C)N3CCC3)CCC2C1 C1(NC(CCCC#C)=O)(CNC(c2cnc(Cl)cc2N)=O)CCCCC1C c1(CC(=O)N(C)CC2CCCN(C(C3C(C=C)C3)=O)C2)nc(F)c(F)cc1F c1(C(=O)NCC2C3CN(C(C(CC)(C)O)=O)CC32)cc(OC)ccc1OC(C)C N#Cc1ccc(-c2cc(NCc3c(Cl)cncc3Cl)ccn2)cc1F C1(C2CCC2)(C(N2C(CNC(c3nn(C)cc3Cl)=O)CC(OC)C2)=O)CC1(F)F Cc1ccnc(O)c1C(N1CCC2(NC(c3ccc(N(C)C)cn3)=O)CC2C1)=O N1(C(C(c2c(F)cccc2F)N(C)C)=O)CCC(C(F)(F)F)C(C)(C)C1 C1(NC(c2c(NC)nc(C)cc2)=O)C2CC(O)C1N(C(C1CCOC1)=O)C2 c1(C(N2CCCC(NC(c3c(C)nccc3)=O)CC2)=O)ncnc2c1cnn2C C(=O)(C(F)(F)C(F)F)N1CC(OCC)(CNC(C23CCCC2C3(F)F)=O)C1 Cc1nccnc1C(=O)N(C)CC=CC(=O)NCC1(F)CCN(C)C1 C12(COC)CC(NC(C3CCCN(C(C)C)C3)=O)(CN1C(C1(C)CC1(F)F)=O)C2 C(=O)(C(C)CN(C(=O)CCc1cn(C)nn1)C)N(CCCOCC)C C1(CN(C(c2nccnc2OC)=O)CC)CCCCN1C(c1nc(O)c(C)s1)=O c1(C(=O)NC2CCCC(C#C)C2)cc(OCCC)c(O)c(OC)c1 c1(CCCC)ccc(C(=O)N(C(C)C2CC2)Cc2nnc(CC)n2C)cc1 CCC(C(=O)NC1(CO)CN(C(C2(C#N)CC3CC3C2)=O)C1)C(F)(F)F c1(C(=O)NC2C=CCN(C(Cc3ccc(C)o3)=O)C2)ccc([N+](=O)[O-])cc1F C1(NC(C2CN(C)CC(C)O2)=O)CCCC12CN(C(=O)CCc1cncs1)C2 C1(O)(CN(C(CC2CC(OC)C2)=O)C)CCN(C(c2cc(C)c[nH]2)=O)CC1 C(CCC(=C)C)(C(=O)N(C1CCN(Cc2ccccc2)C1)C)N(CC=C)CCC CCC(C)C(O)C(C)C(=O)NCc1cn(CC(=O)Nc2cc(C)cc(C)c2O)nn1 CCS(=O)CC(=O)N(CC(=O)NCC(=O)OCC)C(C)C N1(C(Cn2nnc(C)n2)=O)CCN(C(=O)CN2CC=CC2)C(CO)C1 Cc1nc(=N)[nH]c(C)c1C(=O)NCCC1C(C)CCCN1C(=O)CCN(C)CCO N1(C(C2CC(C)C2)=O)CCN(C)C(C(N2C3CSCC2C3)=O)C1 c1(C(N(C2CC(NC(Cn3c(C)ccn3)=O)C2)C)=O)ccc(S(N)(=O)=O)nc1 C(=O)(CC(O)C(C)C)NCc1scc(C(=O)NCC(CC(C)C)OC)c1 C1(CCC)(NC(c2csc(C(F)(F)F)c2)=O)CCCN(C(C2(N(C)C)CC2)=O)C1 c1(C(C(=O)NCCC(=O)OCC)N(CC(=O)NC2CC2)C)csc(SC)n1 c1(C(=O)NC(C2CCN(C(c3nccc(C)n3)=O)C2)(C)C)n[nH]c2ccccc12 C1(CNC(C(C)(O)C2CC2)=O)CC2CCC(C1)N2C(c1cnnn1C1CCC1)=O C(C(C)CC(=O)N1CC(F)(C(=O)N(C(C)CSC)C)C1)OC c1(NCC(C)CN(C)C)cc(=NC2COc3ccc(Br)cc32)[nH]c(C(F)(F)F)n1 C(=O)(C1=CCS(=O)(=O)C1)NCCCCC(C)NC(=O)Cn1nccn1 C1(CCN(C)C(c2sccc2C#N)=O)CCN(C(C2CCC2CF)=O)CC1 c1(CC)nc(C)c(C(=O)NC2CCCCC2CNC(C2SCCS2)=O)o1 c1(C(N(CCCNC(c2n(CC)ncc2)=O)C2CC2)=O)cc(C)c(O)c(C)c1 CC1CN(C(c2cn(-c3ccc(Cl)cc3)nn2)=O)CC1NC(=O)CCC1CCC1 C1(CNC(C(C)CCO)=O)CCCC2(CN(C(C3CN=C4N=CNN4C3)=O)C2)O1 N1(C(C23CC(CCC)(C2)C3)=O)CCC(C)C(CNC(c2ccc(=O)n(C)n2)=O)C1 N1(C(C2C(c3n(C)ncc3)C2)=O)CCCOC(CNC(C2CC2(C)Br)=O)C1 CC1=CCC(N=c2ccnc(N3CCN(CCC(F)(F)F)CC3)[nH]2)CC1 c1(-n2c(C)cnn2)ccc(C(=O)NCCNC(C2COCCO2)=O)cc1 C(CC(C(=O)NC1CC1CC)NC(c1ccc(C)s1)=O)OCC C1(C(=O)NC2C(CC(C)C)C2)COCCN(C(c2nnc(O)cc2O)=O)C1 C1(C(=O)NCCN(C(C)C)CC)(NC(C23CSCC2C3)=O)CC(O)C1 N1(C(c2c(C)nc(C)o2)=O)CCC2(CCCN(C(=O)C(O)C(F)(F)F)C2)CC1 CCC(C(C)C)C(C(=O)NCCOC)N(C1CCS(=O)(=O)C1)CC C(=O)(C1=NOC(C)(C)C1)NCC1CCN(C(CN(C2CCCC2)C)=O)CC1O N1(C(c2cnc(C)[nH]2)=O)CCn2cc(NC(=O)Cc3ccc(O)cc3)nc2C1 OC1CCC(c2nnnn2-c2ccccc2)(NC2CC2c2cncc(Br)c2)CC1 S(=O)(=O)(c1ccnc(S(C)(=O)=O)c1)N1CCCC(C)(CC)C1 c1(CN(C2CC(=O)N(C3CCC(=O)C3C)C2)C(C)=O)cc2ccccc2nc1Cl c1(C(N2CC(CCO)(NC(CCc3scc(C)n3)=O)C2)=O)cc(C)n(C(F)F)n1 c1(C(=O)NC2(C)CN(C(C3CCCO3)=O)C2)nc(Br)c2ccccn12 C1(C(C(=O)N(CC(F)F)CC)C)CCN(C(C2CCN(C)C2C)=O)CC1 N#Cc1ccc(C(=O)NCC(O)CC(=O)NCCCn2nccn2)cc1 C(C)(C(C(C)C)NC(c1cnc(C)n1C(F)F)=O)NC(C1(CC#C)CCCC1)=O C(CC(C)(C)C)(C(=O)NCC1(O)CCCN(C(C2CCC=CCC2)=O)CC1)OC C#Cc1ccc(C(=O)NCC(C2CCOC2)NC(=O)Cc2nnc(S)n2C)cc1 N1(C(CSCC)=O)CCCC(C)(CNC(c2ncc(C)cc2OC)=O)C1 CCCCCC(O)C(C)C(=O)N1CCc2ncn(C)c2C1 Nc1c(F)cc(F)c(F)c1C(N1CC(NC(=O)CCc2cn[nH]c2)CC(O)C1)=O C1(C(N(CCC(=O)OCC)CC=C)=O)CCN(C(=O)Cc2cc[nH]c2)CC1O c1(C(=O)NCC2N(c3nccc(OCC)n3)CCC2C)c(F)ccc(F)c1Cl c12cc(Br)ccc1S(=O)(=O)NN2.c1(C)ccn(C)n1.CC(COC(F)F)N C12(C(=O)NCC3N(c4ncc(C(=O)OC)cc4Cl)CCC3)CCC(C)(CC1)OC2 C(=O)(C1OC(=O)c2ccccc21)NCCCOCCNC(CS(C)(=O)=O)=O N1(C(C(CC(F)F)NC(c2c(C#C)c[nH]n2)=O)=O)CCc2sccc2C1 c1(C(=O)NC(C)C(C)(C)NC(C2CC(C)(F)C2)=O)cnnc(-c2ccccc2)c1 c1(N(CC(CC)C)CC)cc(=NCC(=O)NC2CCCC2)[nH]c(C(F)(F)F)n1 C#CCC(C)(C(=O)NC1CCN(C(C)=O)C1)NC(c1c[nH]c(=NC)s1)=O c1(C2N(C(=O)CC3CCCC3)CCC2)cc(Br)ccc1Cl C1(C)(C(=O)NC2C(NC(C=C(C)C(C)(C)C)=O)CC2)CC(=O)N(C)C1 N1(C(C=C(CC)C)=O)CCC(NC(c2cc(COC)cn2C)=O)C(CC)C1 c1(C(N2CCC(c3cnn[nH]3)C2)C(=O)NCC)ccn(C(F)F)n1 N1(C(C(c2ccccc2)SC)=O)CC2(CC(NC(=O)CCn3ccnn3)CO2)C1 C(C(=O)Nn1cccn1)n1cc(CNC(c2[nH]cc(C(N)=O)c2)=O)nn1 N1(Cc2c(C)cc(C)[nH]2)CC2CCCC(C1)C2C(=O)NC1CCCC(O)C1 C1(C(N2C(C(C)O)CC2)=O)CCCN(C(=O)C(O)C2CCC2)C1 C12(C(N3CCC(NC(c4c(C)n[nH]c4)=O)(CF)C3)=O)CCC(N=[N+]=[N-])C1C2 c1(OC)ccc(C(=O)NCC2(CNC(=O)CC3(C(F)F)CC3)CCOCC2)cc1 C1(CNC(c2nc(CC)sc2)=O)CCN(C(=O)C=Cc2ccccc2F)C1(C)C c1(NC(CCNC(C2(C)CCC(C)CC2)=O)C)ncc(C#N)cc1Cl c1(NC2(CNC(c3ccc(N(C)C)cc3)=O)CC2)nc2cccc(F)c2s1 C1(C)(CNC(C(C2CC2)OCC)=O)CCCN1C(=O)C(=O)C=Cc1cccs1 C1(CCCC)CN(C(=O)Cc2cncnc2O)CCN1C(c1ccnnc1C)=O c1(N2CCCC(O)(CNC(c3c(C)csc3)=O)C2)nccc(S(C)(=O)=O)n1 C(=O)(C1CCc2nccn21)N1CCC(C(=O)N(C2CC3(CC3)C2)C)(CC)C1 CCCC(C(=O)OC)C(=O)NC(CNC(c1ccc(CO)o1)=O)C1CC1 C1(C(=O)NC2C(CC(C)C)CCCC2)CC2(C1)CS(=O)(=O)C2 C12(C(=O)OC)CC(NC(N3CC4(CCCC4)C3)=O)(CCO1)C2.C12=CC=C(C=C1)C2 N1(CC(N2CCC(NC(c3cccn3C(F)F)=O)CC2)=O)CCCCC(O)C1=O c1(OCC)cccc(C(N2CCC(NC(C3COCCO3)=O)C2C)=O)c1N N1(C(C2CC(=C)C2)=O)CC(CNC(C2CCCCS2(=O)=O)=O)CC12CCC2 c1(C(N2CCC(O)(CN(C(CCCCSC)=O)C)C2)=O)cc(C)c2[nH]cnc2c1 C1(NC(C(C)(C)Oc2ccccc2Cl)=O)CC2CC1N(C(C1(C)CCOC1)=O)C2 c1(OCCC)ccc(C(=O)NCC2CCCN(CCC3CCCO3)C2)cc1OC CCC(C)(C(=O)NC1CCC(CCNC(C23CC(CO2)C3)=O)C1)OC C(CN=c1cc(C)c(S(=O)(=O)NC2(CF)CCC2)c[nH]1)(C1CCCC1)OC CC1=CCN(C(C2CC3CC3N2C(=O)C(C)N=[N+]=[N-])=O)CC1 CC(C)C(F)(F)CC(=O)NC1(CCNC(=O)CCCN2C(=O)CCC2=O)CCC1 C1(NC(c2n(CC=C)nnn2)c2ccn(CCC)n2)CCCC(C2CC2)C1 c1(C(=O)NC2C(C)(C)N(C(c3ccncc3F)=O)CC2)ccc2ncnn2c1 CCC(CC)(CO)C(=O)NCC1CCCN(C(=O)COC2CN(C(C)=O)C2)C1 C1(C(C)C)CCCC1(C)NC(=O)COC(C)(C)CNC(=O)CN1CCCCC1C N1(C(C(C(C)C)O)=O)CCCC(O)(CNC(c2[nH]ccc2-c2cccs2)=O)CC1 N1(C(c2ncc(CC)s2)=O)CCN(C(c2cc(Cl)nn2C)=O)CC1CCO N1(C(Cc2c(C)occ2)=O)CCN(C(=O)CC2CCCNC(=O)C2)C(CCO)C1 Cc1cc(F)c(C(=O)NC2CCCCN(C(C3CCCCN3N=O)=O)C2)cc1F c1(C(C(=O)NCCC(=O)OCC)N(C)CCC2CC2)ccc(S(N)(=O)=O)cc1F C=C(C)CC(C(=O)N1CCCC(CC(=O)NC2CCCCC2C(C)C)C1)OC C(N=c1[nH]c(=N)[nH]c(=NC2CCOC3(CCOC3)C2)[nH]1)c1ccc(OCC)cc1 CCCCCCC(F)C(=O)NC(C)(C)CN(C)C(C1(C)CCN(C)C1=O)=O C(=O)(C1=C(SC)CCCC1)NC(CN(C(=O)Cc1scnc1C)CC)C c1(CC2(N(C(N3CC(n4cnnc4)C3)=O)CC3CC3)CCC2)ccccc1 C1(C(=O)NCCn2cc(C(NOCC)=O)nn2)CCCC(F)C1 C1(CNCC(=O)NC2(C)CC2)CCCN1C(=O)OCC CCCCS(=O)(=O)CC(=O)NC(c1nc(C(F)(F)F)no1)C c1(C(N2C(C)CC(NC(CCN(CC)CC)=O)C2)=O)ccn2ccccc12 c1(NCCCCCC)[nH]c(=NCC(C)CC(C)C)nc2c1ncn2C c1(NC(=O)CC2CN(C(c3ccc(Cl)s3)=O)C2)cnc(Cl)c(Br)c1 C1(C(N2CC3(CNC(C4(Cl)CC4)=O)CC2CO3)=O)CCc2nc[nH]c2C1 c1(C(N2C(CCNC(C(c3n(C)ncc3)O)=O)COCC2)=O)cn2c(n1)CCC2 Cc1cc(C(=O)NCCOCCNC(=O)C(c2ccccc2Cl)(C)C)n(C)n1 Cc1c(C(=O)NCC2(CN(C)C(c3c[nH]nc3-c3ccsc3)=O)CC2)ccn1C c1(N2CCC(C)C2)nccc(=NCCOc2cc(F)ccc2F)[nH]1 N1(C(CCCSC)=O)CC(CNC(c2cc(C(N)=O)cn2C)=O)CC(C)C1 c1(C(N2CCC(C(C)(C)NC(CCC=CC)=O)C2)=O)cccc(OC(C)(C)C)c1 N1(C(C2OC3CCC2C3)=O)CCC(N2CCNCC2)CC1 C(CCC(C)C(=O)N1CCC(O)(CNC(c2ccc(OC)cc2OC)=O)C1)OC Cc1nn(C(C)C(=O)NCC2CN(C(C3CC4CCC3O4)=O)C2)c(C)c1[N+](=O)[O-] CCC(C)CC(=O)N1CCC(C(=O)NCC(C)CO)CC1 c1(C(=O)NCC(CNC(=O)CC2COC(=O)C2)OC)cccc(F)c1C#N C=Cc1ccc(NC(=O)NC2(CSC)CCCN(C(=O)OC(C)(C)C)C2)cc1 C#CCCCC(=O)NC1C2CN(C(C3CC3(F)F)=O)CC12 C1(NC(c2csc(-c3ccco3)n2)=O)CC2CN(C(=O)CC3(O)CC3)CC2C1 C(C(O)CCNC(C1CS(=O)(=O)C1)=O)NC(COCC=C)=O C(C(=O)N1CCC(C(=O)NC(c2cccnc2)CC)O1)C1C(CC)C1 c1(CNC(NCCC=CC)=NC)cccc(OCCOC)c1 c1(C(=O)NCC2CCN(C(c3cn(CCCC)nc3C)=O)C2)ccc(F)cc1O c1(C(N2C3CC(CNC(Cc4nnc(C)o4)=O)C2CC3)=O)cc2cccn2cn1 N1(C(CCc2nc(C)c(C)[nH]2)=O)CCC2CN(C(=O)C(C#N)C(C)C)CCC2C1 C1(C(=O)NCCCN(C(c2c(Cl)nn(C)c2Cl)=O)CC)CC(S(C)(=O)=O)C1 C1(NC(c2ccc(C(=O)OC)s2)=O)CCC(NC(=O)CC2CC3COCC23)CC1 N1(C(CC2CC(OC)C2)=O)CC(NC(=O)C=CC2CCCO2)CC1(C)C c1(C(=O)NC2CC(C(=O)Nc3c(C)cc(Br)cc3)C2)n[nH]c2c1CCC2C C1(CNC(C2N(C)CCC2)=O)CCC2(CCN(C(c3cc(F)c[nH]3)=O)CC2)CO1 C1(C(N2CCC(COC)(CNC(=O)CN=S(C)(C)=O)C2)=O)CCc2nnnn2C1 C(N=c1[nH]c(=NC2CC=CC2)[nH]c2c1SCC2)C1(Br)CC1 CC(CCC(=O)NCC1CCCS1)NC(=O)CCC1(C#N)CCC1 C1(C)(C(N2CC(COC)(NC(c3ccnc(OC)c3)=O)C2)=O)CC2CCC2C1 CC(C)(C)CCC(=O)N1CCOCC1CC(=O)NCC(CO)C1CCC1 c1(C(=O)OC)ccc(Cl)c(NC(C2CCCN2C(=O)Nc2cccc(Cl)c2)=O)c1 C(C)(C(=O)NCC1CCC(NC(C2CCCO2)=O)C1)(c1ccccc1)OC N1(C(CNS(N)(=O)=O)=O)CCOC2CN(C(c3cc(Cl)c(F)cc3F)=O)CC12 C1(NC(c2c(C)cco2)=O)CC2CC1CC2C(N1CC(=O)NC(C(C)C)C1)=O c1(OCCC)cccc(-c2cnc(C(=O)NCC(N3CCCC3)=O)nc2)c1 N1(C(c2c(CC)scn2)=O)CCCC(NC(=O)C=Cc2ccnn2CC)C1C CCC(C)CCC(=O)NCc1cc(O)ccc1C C(=O)(C(C(C)(C)C)C1CCCC1)NC1(C)CC(NC(Cc2c(OC)nccc2)=O)C1 C=Cc1cc(C(N2CC(C)CCC2CNC(c2cnsn2)=O)=O)cc(F)c1 C1(CC(N2CCC(N(CCC)C(c3n[nH]cc3Br)=O)C2)=O)C(C)(C)C1(C)C c1(COC(C)C)cc(NC(c2cc(Cl)cn2C)=O)ccc1O C(CCCC(CO)NC(c1ccc(C)cc1)=O)NC(c1c(CC)ncs1)=O N1(C(c2cn(C)nc2C(F)F)=O)CC2(C1)CN(C(C1OCCO1)=O)C2 CC1CC2(CC(NC(C3CN(C(C4CCC(=O)C4)=O)CCN3C)=O)C2)C1 C1(CNC(c2ncn(C)n2)=O)CC12CCN(C(=O)Cc1cc(F)ccc1F)CC2 c1(CCNC(=O)CC2CC2)c(C)csc1C(=O)N(C1CC(CF)C1)C.COC CN1CCC2CN(Cc3ccc(C#N)c(F)c3)CC2C1 C1(CCC(=O)NCC(N2CCCC2)=O)CCCN(C(=O)Cc2cccnc2)C1 C(=O)(C(C(C)(C)C)n1ccnn1)N(CCC(C(C)C)NC(=O)CCN(C)CCO)C Cc1cn2c(C)c(C(=O)NCC3(O)CN(C(=O)C(C4CCOCC4)F)C3)nc2s1 c1(C(=O)OC)ccc2c(c1)OC(CNCCN1CCC(c3nncs3)C1)C2 N1(C(C(C(C)CC)N(C(c2c(CC)c[nH]c2)=O)C)=O)CCOCC(F)(F)C1 C1(CNC(C(C)C)=O)CC2(CO1)CN(C(C1Cn3ccnc3NC1=O)=O)C2 CC(Cc1cnco1)C(=O)NCC(O)CNC(=O)CNc1ccccn1 Cc1ccoc1CNC(=O)C(c1cnn(C)c1)NC(C1CC1C(C)C)=O CCCC(CC)C(=O)N1CCN(C(=O)C=Cc2ccsc2)C(CCO)C1 C1(CC(=O)NC2CC(CC(=O)NCC(C)N(C=O)C(C)C)C2)CCCCCC1 CCCC(CCC)C(=O)NCC(=O)NCC(=O)NC1(C(=O)NC)CC1 c1(C(=O)NCC(CN(C(=O)COCc2nc[nH]n2)C)(C)C)cc(C#N)ccc1Cl C(C)(C)(CC(F)C(=O)NCC(C)C(F)F)NC(c1c(CC)ocn1)=O N1(C(Cn2c(=O)sc(C)c2C)=O)CC(CO)C2(C1)CN(C(C1CCS1(=O)=O)=O)C2 C1(OC)(CNC(=O)Cc2csc(C)n2)CCN(C(c2cc(C(F)F)no2)=O)CC1 c1(C(N2C(CNC(c3ccc(Cl)o3)=O)COCC2)=O)cn2ccsc2n1 C1(CCC)CCCN(C(C2CC(N(C(=O)COC(C)CC)C)C2)=O)CC1 C(C(=O)NCCCC(=O)C1(SCC)CC1)(C1CCCO1)Nc1ccco1.C1(=O)CN1 N1(C(C(CC)C(=O)OC)=O)CCCC2(C1)CN(C(=O)C(=Cc1ccncc1)C)C2 c1(CC(=O)NC2CN(S(Cc3cccc(N(C)C)c3)(=O)=O)C2)ccc(C#N)cc1 N1(C(COCC)=O)CCC2(CCC(CNC(C3CC3C3CCCC3)=O)OC2)CC1 c1(CC)cc(C(=O)NC2COCC2NC(c2ncnn2CC)=O)nn1CCO c1(C(N2C(c3cn(C)nc3)C(=O)NCC2)=O)cc(Br)c2c(c1)OCCO2 C1(c2ccc(C)o2)CCCCN1CC(c1ccc(C(F)(F)F)cc1)O CCCCC(C)CCC(=O)NC(C)(CNC(c1ncc(Cl)cc1Cl)=O)CO c1(CNCC(CO)F)cccc(F)c1I c1(CC(N2C3CCC(C3)C2CNC(=O)C(F)(F)CO)=O)cccc2nsnc12 N1(C(C2(c3ccc(C)cc3C)CC2)=O)CCN(C(=O)CC(=O)N(C)C)CC12CCC2 CCC(C(=O)N1CC(NC(C2(CO)CC2(F)F)=O)C1)OC c1(C(=O)OCC)ccc(NC(=O)CNC(c2ccn(C(C)C)n2)C)cc1C N1(C(CCC(C)SC)=O)CCCC(C)(CNC(C23CC2COC3(C)C)=O)C1 Cc1ccc(C(=O)NC2CCCC(NC(C3(C)CC4CC4C3)=O)C2)cc1Cl C1(CCNC(=O)C(=O)NCc2cccc(N3CCC3=O)c2)CCS(=O)(=O)CC1 N1(C(C2CCCCS2)=O)CC2CC(C1)N(C(c1ccnn3ccnc13)=O)C2 CC1CCC(C(N2CC(C3CCCCO3)C2)=O)N1C(=O)CCc1cnc(O)[nH]1 C1(C(=O)NC2CN(C(C(=Cc3ccncc3)C)=O)CC2C)CCc2nccn2C1 C1(C(=O)N(C)Cc2cn(C(c3ccccc3Cl)C)nn2)(CC)CCCC1O C1(CC(=O)N(C2CCCC2(F)F)C)CN(C(=O)C(C)(C)N2CCCC2)CC12CC2 N1(C(COC(CC)C)=O)CC(C)(NC(=O)Cc2cn(C)cn2)C1 C=CC(CCC)CC(=O)N(CCCCCNC(=O)Cc1c(C)nc(O)nc1C)C CC1CC(=O)NCCN1CCCCC(=O)N(C)C C(=O)(CCCS(N)(=O)=O)NC(C1CN(C(c2n[nH]cc2[N+](=O)[O-])=O)C1)C N1(C(CSCC)=O)CCN(C(c2ccc(N)c(SC)c2)=O)CC1CF CC(C)C(CCN(C)C(C1(CCF)CC1)=O)NC(c1nncn1C)=O Cc1cncc(C(N2CCOCC2CC(=O)NCc2ccns2)=O)c1 CC1(C)CC(NC(=O)C(N2CCCC2COC(c2ccc(Cl)cc2)=O)=O)CCS1 C=CC1(C(=O)Nc2cccnc2)CCN(C(=O)C(=Cc2ccccc2)C)C1 c1(C(=O)NCC(C)(C)OCCNC(C(CC)CCOC)=O)cnn2c1OCCC2 C1(CCNC(CCN(S(C)(=O)=O)C)=O)CCCN(C(C2(C)CC=CC2)=O)C1 c1(C(N2CC(CC(=O)Nc3cc(Br)nc(Br)c3)C2)=O)cc(O)ccc1[N+](=O)[O-] CCCC(CCC)CC(=O)N1CC2CC1C2NC(C1CN(S(C)(=O)=O)C1)=O c1(C(=O)NCc2c[nH]nc2C(N2CC(N3CCCC3)C2)=O)c[nH]c2cnccc12 CC1(C)C(CNC(C2CCCC(=O)O2)=O)CCN1C(c1nccc(Cl)c1F)=O c1(CC(=O)NCCCC2N(C(CC3(OCC)CC3)=O)CCC2)cccnc1Cl c1(C(N(CC(CN(C(C(CC=C)CC)=O)C)O)C)=O)nn(C)c2c1CCC2 c1(C(C)CC(=O)N(C(C)CCNC(c2cncs2)=O)C)ccccc1F c1(C(=O)NC2CC(CC(=O)Nc3ccc(O)c(F)c3)C2)cc2cnccc2[nH]1 Cc1oc(C(C)(C)C)cc1C(=O)N(CCCNC(=O)Cc1cc(Cl)sc1Cl)C CN1CCCC(NC(=O)NC2COCC2NC(=O)COCC2CCCO2)C1 N1(C(=O)NC2CC(C(=O)OC(C)(C)C)OC2)CC2CC2C1C#N CC(CC(F)F)C(=O)N(CCC(N1CCC(F)(CO)C1)=O)CC1CC1 C(=O)(C(C)(C)NC(C)=O)NCC(c1ccccc1)CNC(C(F)=CC)=O CC1C(NC(=O)Cn2cncn2)CCCN1C(=O)CCC(=O)c1ccc[nH]1 CCC(F)(F)CC(=O)NC1CC(CCNC(c2cc(F)cnc2O)=O)C1 C(CCN=C(NCC1CC1)NC1CCC1)N(CCCC)C CN1CCCC(N=c2[nH]c(=N)[nH]c(=NCC3CC3C3CCOCC3)[nH]2)C1 N1(C(c2c(C)cnnc2O)=O)C2CCC1CN(C(=O)COC1CC1(F)F)C2 c1(CC(=O)N(CC(O)CNC(C2CCCC2CF)=O)CC)nn(C)cc1Cl N1(C(C2(O)CCCN(C(=O)OC)C2)=O)CCCC12CCCN(C(=O)CSC)C2 c1(C(N(C2CCN(C(C3CC(C)C3)=O)C2)CCO)=O)cc(C#N)ccc1O CC1(C)COc2cc(NC(c3nnnn3CCC3CC3)c3cn[nH]c3)ccc21 O=C(C1=CC2(CCN(C(=O)C(O)Cn3cncn3)C2)C1)NCc1ccc(O)cc1 N1(C(c2c(C)cc(CC)o2)=O)CC(C(N2CCC=CC2CC)=O)CCC1(C)C N1(C(CC(C)OC)=O)C2COCC1CC(NC(=O)CN(C)Cc1ccccc1)C2 C(=O)(CC(C)c1cnn(C)c1)NC(CC)CN(C)C(C1CC(N2CCCC2)C1)=O C=CC1(CC(=O)NCC(=O)N(C)OC)CN(C(c2ccsn2)=O)C1 C1(CC(=O)NC(CCN(C(=O)CSc2nc[nH]n2)C)(C)C)CCC(=O)NC1 c1(OC)ccnc(CNC(=O)CCC2CCCN2C(C2C(C)C2C)=O)c1 c1(C(=O)NCC2CC(NC(CC3C(C)(C)COC3)=O)C2)cnc2[nH]ccnc1-2 CCC(C)(CCC(C)C)C(=O)NC12CCCC1N(C(=O)CNS(C)(=O)=O)CC2 c1(C(=O)NC2CN(C(C(CC#C)O)=O)CC(C)(C)C2)cnc(O)c2ccccc12 Cc1oc(C2CC2)nc1C(=O)NC1C=CC(CNC(C2CC3CCC2O3)=O)C1 C(C(C)(C)C(C)(C)O)NC(C=CC1N(C(c2nc(CC)oc2C)=O)CCC1)=O c1(C(=O)NCC2CCC(C)N(C(c3cc(C)n(C)n3)=O)C2)cc(F)c(F)cc1O c1(NC(C2CC(NC(C(c3ccccc3)C)=O)C2)=O)cnc(Cl)nc1 c1(C(=O)OC)ccc(Cn2ccc(C(F)(F)F)n2)cc1.C1(C)CC(=O)N1 C1(CC(N2CC(O)(COC)C2)=O)CN(C(c2cc(OC)cs2)=O)CCC1C C1(CNC2C(CC)N(C(=O)OC(C)(C)C)C2)Cc2cc(Br)ccc2O1 CC(F)C(C(=O)N1CCCC(NC(c2ccc(Cl)o2)=O)C1)NC(=O)OC(C)(C)C c1(C(N2CCC(NC(C(C(C)C)C)=O)C23CCC3)=O)ccc2ncncc2c1 N1(C(C(CC)(C)C)=O)CCN(C)C(C(N2C(CO)CC2C)=O)C1 c1(SC)cc(C(N2CC(CCNC(c3ccc(O)cn3)=O)C2)=O)ccc1F C1(OCC)CCC(n2cc(C(C)N(C(=O)C(c3ccc(C)cc3)O)C)nn2)CC1 C(CCN=c1c(C#N)c[nH]c2cc(F)cc(F)c12)N(C)C(C1(C)C=CCCC1)=O CC1(C)C(CNC(=O)C(=O)Nc2ncc[nH]2)CCN1C(=O)CC1CCCCC1 N1(C(c2c(C)cns2)=O)CC2CCN(C(C3CN=C4N=CNN4C3)=O)C2C1 N1(C(Cn2c(C(C)C)ncc2)=O)CCC(C)C(CNC(C23CC(C)(C2)C3)=O)C1 C1(C)(C(=O)NCC(C)(C2CCC2)NC(=O)C(C)(C)n2cccn2)C=CCC1 c1(CNC(c2nc(C)c(C)n2C)c2n(C(CC)C)nnn2)cn(C)c(=O)nc1O CCCCC(C(=O)NCc1ccc(C2CC2)o1)NC(=O)C(F)C1CCCC1 C1(NC(c2ccc(CF)cc2)=O)CN(C(=O)C=C2CCC2)C2(CCOC2)C1 C1(C(=O)NC(CCC)c2ccco2)CC(CC)CCN1C(=O)CCS(N)(=O)=O c1(OC)cc(C(N2CCC2CNC(=O)CC2CCCC2)=O)cc(F)n1 C1(N(CC(=O)N(CCCN(C)C)C)C)CCN(Cc2c[nH]nc2C(C)(C)C)CC1 c1(OC)ccc(NC(=O)C(C)NC(C2COC(=O)N2C)=O)cc1C C=C(C)CCC(=O)N1CC2C(CN(C)C(C3CC3c3cncs3)=O)C2C1 S(=O)(=O)(c1cccnc1NCc1ncoc1C(F)F)NCC(CC)(CC)SC N1(C(C(CCNC(C2CC(CC3CC3)C2)=O)OC)=O)CCOC(C)(C2CC2)C1 C12(C(N(CC(CNC(C(CC)(F)F)=O)O)C)=O)CCC(CC1)C2(C)C N1(C(CC(C(=C)C)OCC)=O)CCC2(C1)CN(C(c1c[nH]cc1C)=O)CCO2 c1(CC)cccc(F)c1NC(=O)CC1CCCCN1C(=O)CSCC(F)F CC(CC(=O)N1CC(CNC(c2cn(C)[nH]c2=N)=O)C(C)(C)C1)C(F)(F)F C1(NC(C(C(C)NC(c2ccsc2)=O)C)=O)CC2C(O)C(O)CC12 C(=O)(C1CCCc2cccnc21)NC(CNC(=O)CC1(O)CCCCC1)CO C1(CNC(C2C(CC)C2)=O)CCCN(C(=O)CCC2CC2)CC1 c1(C(=O)NCC(C2CC2)NC(c2cc(Cl)cnc2O)=O)cc(F)cnc1O N1(C(C2CCC(CC)O2)=O)CCC(NC(=O)CCn2ccc(C)n2)CC1C C1(CNC(C(C)=C2CC2)=O)CCCN1C(=O)C=Cc1cn[nH]c1 Cc1ccc(F)c(C(=O)NC(C)C(=O)NC(c2cccnc2)CO)n1 CCC(C)(C#N)C(=O)NCC(O)CNC(=O)Cc1ccnc(C)c1 N1(C(c2cc(C)ns2)=O)CCCN(C(=O)COCC2CCCOC2)C(C(C)C)C1 C(=O)(CCCC(=O)C(C)(C)C)N1CC(C(C)C)N(C(c2nn(C)cc2Cl)=O)CC1 N1(C(C(CC#C)(C)NC(c2ccc(=O)n(C)c2)=O)=O)CCC2(CCC2)C(O)C1 c1(C(=O)NCC2(CNC(=O)Cc3ccsc3)CC2)cnc(-c2ccccc2)o1 C(=O)(C(CNC(c1ccsn1)=O)CC(C)C)NCc1c(CC)onc1C C1(CC(=O)NC(C)CN(C)C(c2cc(C(N)=O)no2)=O)CC2(CCC2)CCO1 N1(C(c2c(CC)ocn2)=O)CC2CC2(NC(c2cn(C)nc2-c2ccoc2)=O)C1 C12(NC(Cn3ccc(C)n3)=O)CCOCC1CN(C(c1[nH]c(C)cc1C)=O)C2 C1(CC)COC(C)(C)CN1C(C1CN(C(=O)CCc2cncs2)CC(C)O1)=O N1(C(CC2CC(=C)C2)=O)CC(NC(=O)C(C)(C)F)C(C)C1 NC(=O)CCCCC(=O)NCCCC1CCCN1C(=O)CCS(N)(=O)=O CC(C)CCC(=O)OC1COC1.N1(C)CCN(C(c2ccccc2O)=O)CC1 N1(C(C(CC)C)=O)CC2CCC(CNC(c3ncc(F)c(OC)n3)=O)(C2)C1 N1(C(c2cc(C)[nH]n2)=O)CCC2CCN(C(c3cc4c(C)n[nH]c4cn3)=O)C2C1 c1(C(N2CCN(C(C3=CC(C)(CC)C3)=O)CC2)=O)ccc2occc2c1 c1(OC)ccc(C(=O)NCC(c2ccc(C)cc2)NC(=O)COC2CC2)c(F)c1 N(C(=NCCCOC(F)(F)F)NC1CC12CCC2)C(c1ccccc1)C1CC(F)C1 C(C(F)(F)CCC(=O)NC(c1cc(Br)no1)C)n1cc(CCCC)nn1 CC1(C)CC2CN(C(C3CCN(C(=O)c4nnsc4N)O3)=O)CC12 c1(C(CNC(=S)NCC23CC(CCO2)C3)C(F)(F)F)c[nH]c2ccccc12 N1(C(=O)NC(c2ncc(-c3ccccc3)[nH]2)C(C)C)CC(F)C(F)C1 C(CC(C(C)C)NC(=O)Cc1csc(NC=O)n1)NC(CC(=C)C)=O S(=O)(=O)(c1ccc(CCN2CCC(O)C2)c(F)c1)N(CC(C)O)CCC1CC1 C1(NC(C=C(C)C)=O)CN(C(c2cnc(C)nc2C)=O)C2(CCCC2)C1 N1(C(C2(C)CNC(=O)C2)=O)CC2CC(C1)N2C(C1(F)CCCCC1)=O c1(CC(N2CC(CC=C)(NC(C3COC(=O)O3)=O)C2)=O)ccccc1Br C(C(=O)N=c1cco[nH]1)N1CC(CN(C)C(c2ccnc(F)c2F)=O)C1 C1(OCCCC(=O)NCCN(C(C2C(CCC)C2)=O)CCC)CCC(C)CC1 C1(C)(C(=O)NCCN(C(C(COC)C)=O)CC(C)O)CCCN(C)C1 c1(C(=O)NC2C3(CN(C(C4CC(SC)C4)=O)C3)CC2)cc(C)c(C)nc1C Cc1cc(C(N2CCC(C)(C)C2CNC(=O)CC2CCN(C)C2)=O)cc(C)c1 C1(CN(c2ccnc(NCCCC(C)O)n2)C)Cc2ccccc2CO1 C(=O)(C(CC(C)(C)C)OC)N(C(C)C(=O)NCCCN1CCOCC1)CC C1(CC(=O)NC(c2ccc(-n3c(C)cnc3O)cc2)C)CCC2CNCCC2C1 C=CCCCCC(=O)NC1(CCOC)CCN(C(C2OCCOC2C)=O)CC1 Cc1sc(O)nc1C(=O)NCC1(F)CCN(C(=O)CC2CC2C2CC2)C1 C1(C(=O)NC(CNC(c2ccnc3cc[nH]c23)=O)CO)Cc2cc(Cl)ccc2O1 C1(CC(=O)NC2(CC)CN(C(C3C4CCCC34)=O)C2)CCN(C)C1=O Cc1ccc2scc(C(=O)N(CCCNC(=O)CC(C)(C)c3cccs3)C)c2c1 N1(C(C(N2CC(C)OC(CO)C2)=O)=O)CC2CCCN2CC1C(=O)O c1(C(N2CC(NC(C3CC4(C3)CC(F)C4)=O)C3(C2)CC3)=O)cc2ccccc2o1 c1(CN(CC(C)C)C(=O)NCC2(C)CSC2)nocn1 c1(C(N2CC(COC)(CNC(=O)CCN3CCC3)C2)=O)nc(OC)cc(OC)n1 C1(N(C)C)CN(C(C2CCCN2C(=O)CCCn2ccnn2)=O)CC1(C)C C1(CNC(C(c2cccc(C)c2)O)=O)CCN(C(c2ccnc(C)n2)=O)C(C)C1 C1(C(=O)NCC(CN(C)C(C2(CO)CC2(F)F)=O)(C)C)C2CCCCC12 C(=O)(CC(C)CCC(=O)NCCCCCCNC(=O)CC(=O)NC1CC1)OC c1(C(=O)NCCC(=C)CNC(=O)C(C)CF)cnc(C)c2c1COC(C)(C)O2 c1(C(N2CCN(C(C3CC(CC)C3)=O)CC(O)C2)=O)ncnc2c1ccn2C c1(NC(C2CCCO2)C)ccc(S(=O)(=O)NCc2cnc3n2CCCC3)cc1Cl c1(C(N(CC(CC)NC(c2oncc2C)=O)CC)=O)ccc(OC2CC2)cc1F N(C(=NCCN1CCCCCC1)NCC1(C)CCOC1)C(CC)C C1(NC(=O)NC(COC)C(C)(C)O)CN(C(=O)OC(C)(C)C)CC1O C(=O)(C(C)(C)CC(=O)NC(Cn1cncn1)C(=O)NCC(CO)N(C)C)OC N1(C(C(CC=CC)C)=O)CCCC(C)(C)C1CNC(=O)CC1CC(C(=O)OC)C1 CCC(CC(=O)NC(c1nccc(C)n1)C)N(C(=O)Cc1cccnc1OC)C C(=O)(C(CCC(N)=O)n1cc(CC2CCCCC2)nn1)NC1C(C)C1(C)C N1(C(Cc2scc(C)c2)=O)CCC2(CCN(C(c3cccc(C)c3C)=O)CC2)C1 C=CCC(C)(C)CC(=O)N1CC(N(C(=O)CC(C)(C)SC)C)C1 N1(C(CC(=C=C)C)=O)CC2(CC(C(N3CC4CC5CC4C3C5)=O)CO2)C1 C1(CNC(C=C(C)C(C)C)=O)(NC(=O)C(F)CC2CCC2)CCCC1 CC(C(C)(C)NC(=O)C=Cc1cscn1)NC(c1cc(Cl)no1)=O N1(C(c2n[nH]c(C)c2C)=O)C2CCC1C(CNC(c1ccc(Br)cc1)=O)C2 N1(C(CCCCC)=O)CCOC2(CCN(C(=O)CCc3cccnc3C)CC2)C1 CCC(CC(=O)N1CC(CC(C)NC(c2cccc(C(C)(C)C)c2)=O)C1)C(F)F c1(OC)ccc(C(=O)NCC2CCN2C(=O)CCCN(C)C(C)=O)c(F)c1 c1(SCC)cc(C(=O)NCC2CCCN2C(=O)C(C)C2CCC2)ccn1 Cc1ccc(CN2CC(NC(C3CCCN(C(=O)C4CC4)C3)=O)C2)c(F)c1F C1(C(N2CC(CC)(NC(=O)C(C)CC#N)C2)=O)CCCC(N(C)C)C1 C1(NC(C2C(C(=O)OC)C2)=O)CC(N(C(=O)CCn2cncn2)C)C1 C1(C(N2CC(CNC(C(C)(C)N(C)C)=O)CC2(C)C)=O)CCc2ccnn2C1 c1(C(=O)NC2CN(C(C3=CCCCC3C)=O)C2)c[nH]c2cccc(C#N)c12 C1(OC)CC(CNC(=O)Cc2nnc(C)o2)N(C(C2(c3cc[nH]n3)CC2)=O)C1 Cn1ncc(C(=O)NC2CC2NC(c2ccc(-c3ncc[nH]3)cc2)=O)c1N C1(CNC(C2=CCSC2)c2n(-c3c(Cl)cccc3)nnn2)C2(CCC2)C12CCC2 N#Cc1c(N2CCCC(CCNC(c3cc(CO)[nH]n3)=O)C2)ncc2c1CCC2 C1(NC(c2[nH]c(CC)c(Cl)n2)=O)CC(OC)CN(C(C2CCCSC2)=O)C1 Cc1ccc(C(=O)NCC(O)CNC(=O)CC2CC3CCC2C3)nn1 c1(C(=O)NCCC2CC(NC(Cn3ncc(C#C)c3)=O)C2)cccc2nncn12 CCC(C)(C(=O)N1CC(C2CN(C(c3coc(C4CCC4)n3)=O)C2)C1)C(N)=O C(=O)(C1=NOC(C(N2CC(=C(F)CNC(C3(CO)CCOCC3)=O)C2)=O)C1)OC C(=O)(C(O)C(F)(F)F)NCC(C(=O)N(CC(CCC)C)C)N(C)C c1(C(=O)NC2CC(NC(C3N(C(C)=O)CCC3)=O)C2)c(C)ccc2nonc12 C(C)(C(CC(=O)N(C)Cc1cncs1)NC(C1(OC)CCSC1)=O)OC C(CC(O)CC(=O)NCC1(C)CCCN(C(=O)C(F)C(C)(C)O)C1)SC C(=O)(CC1=NNC(=O)C1)N1CC(O)(CCNC(c2cccc(C)c2F)=O)C1 C(c1cc(C)c(C)cc1C)=CC(N1C(C(=O)OC)CCC(C(=O)O)C1)=O c1(NC(C2C=CC(C(=O)NC(COC)C)C2)=O)ccccc1SC(F)F CCCC(CCC)C(=O)N1CCCC1CC(=O)Nc1cccc(I)c1 c1(C(=O)NC(C)CNC(C2(C)CC=CCC2)=O)cnn2c1NCC(C)C2 Cc1ccc2sc(C(=O)NC3CCN(C(c4cn(C)nn4)=O)CC3(C)C)cc2c1 c1(OC)ccc(C(=O)NC2(c3nn[nH]n3)CCC2)cc1[N+](=O)[O-] c1(-c2cc(C(=O)NC(c3ccc(C)o3)C)no2)ccc(F)cc1F c1(C(=O)NCC2(F)CC(NC(C3(C)CCOC3)=O)C2)ccnc(CO)c1 C1(NC(c2c(C)ocn2)=O)CN(c2ncc([N+](=O)[O-])cc2Br)C2CCCCC12 CC(C)(CC(F)F)C(=O)N1CCCC(O)(CNC(=O)CCC2=CCCC2)C1 CC(C)CC(C)C(=O)N1CC(N(C)C)C(CNC(=O)COC2CCCC(C)C2)C1 c1(C(=O)NCC2N(C(c3n(C(CC)C)ncc3)=O)CC=C2)c(OC)cccc1F c1(OC)nc(C(F)(F)F)ccc1NC(C1CC(F)CN1C(=O)C(C)(C)Br)=O C1(C(=O)NCC23CC(NC(c4cccc(NC)n4)=O)(C2)C3)CC1C1CCCC1 C1(C(N(C2CC(C#N)C2)CC(=O)NC(C)(C)CC2CCOC2)=O)CCC(=O)NC1 CC1CCC(NC(=O)C=CCN2CCC2)CN1C(C1CC2(CSC2)C1)=O N1(C(c2cc(OC)c(Cl)s2)=O)CC(C2CCCCN(C(C3CC3F)=O)C2)C1 N1(C(c2cn(CC)nc2)=O)CC(NC(=O)CC2CCC(C)O2)C(CC(C)(C)C)C1 C1(NC(C(C(=O)OCC)OC)=O)CN(C(=O)CCS(=O)(=O)NC)C2(CCC2)C1 Cc1cnncc1CNC=O.C12(CC1)C(=O)N2 c1(CC(N2CCN(CCN(C(CCC#C)=O)C)CC2)=O)c[nH]c2cc(F)ccc12 C1(CNC(CN(C)CC)=O)COC(C)(C)CN1C(C1CC1(C)C(F)(F)F)=O Cc1cc(O)n2ncc(C(=O)NC34CCCC3N(C(=O)C(C)CF)CCC4)c2n1 C1(NC(c2nc(C)sc2C)=O)CC(CNC(c2cn(C)cn2)=O)C12CCC2 Cc1nc(C(N2CC(C3CN(C(=O)Cn4cnnn4)CCO3)C2)=O)sc1C n1(CCC)cc(C(=O)NC(C2(O)CN(C(=O)CSCC)C2)C)cn1 C(=O)(CC(C(F)(F)F)NC(C1CC(=O)CC(=O)N1)=O)NC(c1n(CC)ncn1)C C1(CC(=O)NCCN(C(c2cnn(C)n2)=O)CC)Cc2ccccc2NC1=O c1(C(N2CC3CC3(C(=O)Nc3ncc(I)cn3)C2)=O)cc2ncccc2[nH]1 C1(C(=O)NCC2CCCN(C(C(CC)C)=O)CC2)CC2(C1)CC1(CC1)C2 N1(C(CC(CC)OC)=O)CCN(C(c2coc(C(F)(F)F)n2)=O)CCC1C C1(CNC(C2(CC=C)CN(C(c3cnsc3C)=O)C2)=O)CCCCC1C c1(C(=O)NC2C(NC(CC3(COC)CCOCC3)=O)C2)cc2cccnc2[nH]1 C1(C)(C(=O)NC(CN(C(CSCCC)=O)C)C)CC(C(C)C)=NO1 CCCC(CCC)C(=O)NCC1CCCC1C(N1CCC(F)(C(=O)OC)C1)=O C(=O)(C1=CC2C=CC(C1)C2)N(CC(C)CNC(=O)Cc1ccc(C(F)F)cc1)C C=C(Cl)CC(C(=O)N(C1CC(O)C1)C)NC(C1CCC1C#N)=O c1(NC(=O)CC2CC(CF)C2)ccc(NC(=O)Cn2cc(Br)cn2)cc1F c1(CCC)cccc(C(N2CCC(OCCNC(=O)C=C3CCCC3)C2)=O)c1 C1(NC(=O)C(N2CCC(CC(F)F)C2)=O)CCCC(C(F)(F)F)C1 c1(C(=O)NCCCC(C)NC(C2(OC)CCOC2)=O)cccc(F)c1O N1(S(C)(=O)=O)CCCc2cc(-c3nc(-c4ccncn4)no3)ccc21 N1(c2ccnc(C(CC)C)n2)CC2CCC(NC(=O)CS(N)(=O)=O)CC2C1 C(=O)(C(=O)N(O)C(C)C)NCC(CNC(c1cnc(N(C)C)c(Cl)c1)=O)C N1(C(=O)OC(C)(C)C)CCCOC(CNC(c2ccnc(F)c2O)=O)C1 CC1(C)CC(C(=O)NCC2(C(C)(C)C)CCN(c3ncccn3)C2)CC(C)(C)C1 c1(-c2scc(-c3nc(CC4(CC)CC4)nn3C3CCC3)n2)ccc([N+](=O)[O-])cc1 N1(C(C(C2CCOC2)NC(COCC)=O)=O)CC(C)C(O)C1 c1(C(N2CCCN(C(c3onc(C)c3C)=O)C(C)C2)=O)c(F)ccc2ccoc12 N1(C(C=CC)=O)CCN(C(c2cnn(C(C)C)c2C)=O)C(C(F)F)C1 Cc1cc(C(N2CCC(CNC(c3cnc(S)nc3)=O)CC2)=O)cc(C)n1 C=CCCN=C(NCc1ccn(C)c1)NC1CC(=O)N(CCN(C)C)C1 C1(O)(CCNC(CCC=C(C)C)=O)CCN(C(=O)CCn2ccnn2)CC1 C1(CCO)(NC(C2C(C)C2)=O)CN(C(c2cn(C)cn2)=O)C1 C12(COCC(=O)NCCNC(CCN(C)C(c3nc[nH]n3)=O)=O)CCCC1C2 CCCC(C)C(=O)NC(c1ccccc1)CNC(=O)C(N)=O N1(C(CN(C2CC2)CC)=O)CCCCCCC1C(=O)NCc1ccnc(F)c1 O=C(C1=CCOC1)NC1CN(C(C23CC(O)C2C3)=O)CC1O c1(NC(c2n(CCOCC)nnn2)c2ccc(OC)o2)cccc2nc[nH]c12 c1(C(C)(C)C)nnc(Cn2cc(CNCCCO)nn2)s1 c1(N2CCC(F)(CNC(c3cccc(N(C)C)n3)=O)CC2)nc(C#N)ncc1Cl c1(CN2CCN(C(C=CC)=O)C3C2C3)cc(OC)c(OC)c(F)c1 C1(C(=O)OCC2CC(COC)C2)CC12CCOc1ccccc12 CCC(CN=c1cc[nH]c(=NCC)[nH]1)c1ccc(C#N)cc1.N(C)C C1(NC(C(C)(C)c2ccno2)=O)CCN(C(c2ccc(CO)o2)=O)C12CCC2 C(=O)(C(CC(C)C)n1ccnc1)N1CCC(C(CNC(CNC(C)=O)=O)C)CC1 Cc1nccc2c1CCN(C(c1ccc(F)c(Br)n1)C(=O)NCCC1CC1)C2 c1(C(=O)NC(CC(C)NC(c2coc(C(F)F)n2)=O)C)ccc2cccnc2n1 C(=O)(CCC(C)(C)F)N1CCC(OCCNC(C2C(C)OCC2)=O)CC1 C1(N(C(C(C)Cc2cccnc2)=O)C)CN(C(=O)C=Cc2ncco2)CC12CC2 C1(C)(N(C)C)CCN(C(c2cc(CNC(C3CN(C4COC4)C3)=O)on2)=O)C1 N1(C(COC(C)(C)C)=O)CCC(OCC(=O)NC2CCNC(=O)C2)C2CCC12 Cc1cnccc1C(=O)NCCCCN(C(=O)C(C)SCC1CCCO1)C c1(N(C)Cc2ncc(C)nc2)nc(=NC2CCC(F)CC2)[nH]c2ccccc12 C(=O)(CCCCC(F)(F)F)NC1(CCNC(C2N(C=O)CCC2)=O)CCC1 c1(C(N2CCC(N(C(=O)Cn3nnc(=O)[nH]3)CC)C2)=O)noc2c1CC(C)CC2 C1(CO)COCCN(c2nnnn2Cc2nc(C3CCOCC3)n[nH]2)C1 c1(CNC2CC(C)(C(C)(C)C)C2)cc(C(F)(F)F)cc(Cl)n1 C(=O)(C1=NN(CC)C(=O)CC1)N(C1CCN(C(C2C(=C)CC2)=O)C1)CC Cc1nccn1CC(=O)NC1CC(C)(CNC(=O)CC2CC2)C1 c1(C(C(N2CCC(CN(C(C(C(C)C)SC)=O)C)CC2)=O)O)c(C)cccc1C C1(NC(C(C)OCCOC)=O)CCN(C(C2CCC(OC)CC2)=O)C12CC2 C(=O)(C(C)(C)CF)NC(C)C.C(=O)(C(=O)NC)N(CCNCC)CC N1(C(CC(CCCCC)O)=O)CC23CCCC2(C1)CN(C(=O)CN1CC=CC1)C3 CCCC(C)(C)CC(=O)NCC(C1CCOC1)NC(=O)CCC1(CC2CC2)CC1 c1(C(N2C(C3(NC(CCSCC)=O)CC3)CCCC2)=O)ccn(C(C)C)c(=O)c1 C(C)(C(=O)N(CCC(=O)N1CCC1CO)CCCO)NC(CCCC)=O c1(NC(CNC(C(=O)OC(C)(C)C)CC#N)=O)ccc(F)c(Cl)c1 CCCCCC(O)CC(=O)NC(C)(CSC)C(=O)NC(c1ccc(C)cc1)C c1(C(N2C3CN(C(CCS(=O)(=O)NC)=O)C(CC3)C2)=O)c(C)nc2sc(C)nn12 c1(C(=O)OC)cc(Br)ncc1NC(=O)CC1(C)CN(Cc2ccnc(Cl)c2Cl)C1 c1(C(N(C(C)CNC(=O)Cc2cc(F)ccc2Cl)C)=O)cc(Cl)c(F)cc1F C1(NC(C(C)SC)=O)CCCCCN(C(c2csc(C)c2Br)=O)C1 C1(C(=O)NC2CCC(NC(CCNC(N)=O)=O)C2)CCCS(=O)(=O)C1 c1(C(N2CCC(O)(C(F)(F)F)C2)=O)cc(C(F)(F)F)nc(C2CC2)c1 C1(NC(=O)C(C2(O)CN(C(=O)C(F)(F)C3CC3)C2)F)CCCCC1O c1(C(=O)NC2CC(C)(NC(c3nn(C)c(O)c3)=O)C2)ccc(S(=O)CC#N)cc1 Cc1ccc(=O)n(CC(N2CCC(NC(c3c(C)cncc3C)=O)C(F)C2)=O)n1 C1(O)(CCNC(c2cnc(C(F)F)s2)=O)CN(C(C2C3CCCC23)=O)C1 C(C)(C)(C(=O)N1CC(O)CCO1)C1CCN(C(C(C)OCCC(C)C)=O)C1 c1(C(C(=O)NCCC)N(C2CCCC(P(C)(C)=O)C2)C)cc(F)cc([N+](=O)[O-])c1 Cc1cc(C(=O)NCCCCN(C)C(c2c[nH]nc2I)=O)n[nH]1 N1(C(c2cc(CC)on2)=O)CCCC2(NC(c3ccccc3OC)=O)CC12 c1(C(N2CC(N(C(Cc3nnc(C)s3)=O)C)C2)=O)cc(CN(C)C)ccn1 C1(CC(=O)N(CCC)Cc2cn(C(C)C(=O)O)nn2)CCC(F)(F)CC1 CCCC(C)(O)CC(=O)NCC1(NC(c2ncc(Br)cc2C)=O)CCC1 c1(N2CCC(CC(C)NC(CNC(=O)NC)=O)CC2)ncc(Br)c(O)n1 N1(C(=O)Cn2nccn2)CC2CC1CN2C(c1cc(C2CC2)ns1)=O C1(CNC(Cc2ccn(CC)n2)=O)CCCN(C(C2CCC(C)O2)=O)C1 C(=O)(CC(C(F)(F)F)N(C)C1CC1)NCC1=CCN(C(C(C=C=C)C)=O)CC1 c1(CCC(=O)N2CCC2Cn2ccc(C(=O)O)n2)nc(-c2cccs2)no1 c1(CC)nn(C)c(C(=O)N(C)CCNC(c2ocnc2C2CC2)=O)c1Cl N1(C(c2noc(C)c2C)=O)CCN(C(c2cc(Br)ccc2Cl)=O)C(C(C)C)C1 C(CCCCCCC(F)(F)F)N1C(CC(C)C)CC(O)C1 N1(C(CCC2CC(C)C2)=O)CCCC1C(C)NC(c1nccn1C)=O C1(C(=O)NC(CC)CCCO)CCCN(C(=O)CC2CSCCO2)CC1 N1(C(c2nnn(C)n2)=O)CCC2CN(C(c3c[nH]cc(Br)c3=O)=O)CC2C1 CC1(NC(=O)NCc2ncco2)COC(C)(C)OC1 c1(C(=O)NCC2CC(=C)C2)nc(O)c(C#N)cc1C CCCCCCCCOCC(N1CCC(NC(c2snnc2C2CC2)=O)C1C)=O S(=O)(=O)(c1cc(C)cnc1N1CCC(c2ccncn2)CC1)N(CC)CC1CC1 N1(CC=C)CCC(NC(=O)C(CCF)NC(=O)CC2CCC(=O)C2C)CC1 c1(OCC(=O)NC(C)C(C)NC(=O)Cn2cccnc2=O)cncc(Br)c1 CS(=O)(=O)c1ccc(CC(CC(=O)NCCBr)NS(=O)(=O)c2cccc(Cl)n2)cc1 C12(NC(=O)CCc3cnoc3)CC(CNC(C3CC=CC3)=O)(C1)C2 Cc1nnc2n1CC(C(=O)NC13CC(NC(=O)CC4(CO)CC4)(C1)C3)C2 C1(C(=O)OC(C)(C)C)(CC)CCN(C(N(C)Cc2cn(CC(CC)O)nn2)=O)C1 CCC(CC)C(O)CNC(c1csc(CNC(C2CCN(C)CC2)=O)c1)=O N1(C(C(C(C)c2ccccc2)O)=O)CCCCC12CN(C(c1csc(=N)[nH]1)=O)C2 c1(C(C)NC(C2CC(N(C)C)C2)=O)nc(C(=O)NCC(O)CS(C)(=O)=O)co1 c1(C(=O)NCC2N(C(COCC(=O)NC)=O)CCC2)ccc(F)c(C)c1Cl c1(C(=O)NCC(C)(C2CC2)NC(C2CC3CC3C2)=O)ccc2ccnn2c1 c1(CC(=O)N(CCn2cc(CNC(=O)CC#N)nn2)CC)ccc2c[nH]nc2c1 Cn1nc2c(c1C(N1CC(C3(NC(=O)Cc4cccnc4)CC3)C1)=O)CCC2 c1(C(=O)NC2CC2C(=O)NCCn2cc(Br)cn2)cc(Cl)c(Br)c(Cl)c1 C12CC(C)(C1)NC2=O.C1(NC(C=CC(=O)OC(C)(C)C)=O)CC(C)(CO)C1 N1(C(C2CC(=C)C2)=O)CC(C2CCCCN(C(=O)CCC3C(=O)ON=C3C)C2)C1 C1(C(=O)NCc2ccc(OC)nc2)CN(Cc2ccc(C)cc2Cl)CCC1O c1(CC(N2CC(CCCCNC(CNS(CC)(=O)=O)=O)C2)=O)c(C)nn(C)c1Cl Cc1c(C(=O)NC(C2(O)CN(C(C3CC(F)C3)=O)C2)C)ncn1C CCCCC(CN(C)C(C1(C(C)NC(=O)Cc2cncc(O)c2)CC1)=O)CC N1(C(C2=C(C#N)CCC2)=O)CCC2CCN(C(c3cc4ccncc4o3)=O)C2C1 Cc1cnc(C(=O)NCC2(O)CCCN(C(=O)Cc3nc[nH]n3)C2)cc1Cl C1(N(C(Cn2nnc(C)n2)=O)C)CN(C(=O)COCCN(C)C)CC12CC2 c1(C(=O)NCCCC(C)NC(c2ccc(CO)o2)=O)n[nH]c2c1CS(=O)(=O)CC2 CCN=c1[nH]c(C)c(C(=O)NC2CC2NC(=O)Cn2cc(C3CC3)nn2)s1 C1(N(CCC)C(c2ncoc2CC)=O)CCN(C(=O)Cc2ccon2)CC1 N1(C(CNC(CCC)=O)=O)CCC2(C)CN(C(=O)CCC(CC)CC)CC12 c1(C(=O)NCC(C)=CC(=O)NCC(N)=O)cc(C)ncc1C N1(C(c2c(Cl)cn(CC)n2)=O)CC(CNC(c2cnc(OC)nc2)=O)CC1(C)C C1(OC)CCC2(C(N3CCC(CCNC(=O)C(c4ccccc4)F)CC3)=O)CC12 Cc1nc2cc(C(N3CCCC(CNC(=O)CC4C(C)C4(F)F)C3)=O)cnc2[nH]1 N1(C(CC(=O)NCC)=O)CCC(CN(C(=O)C(c2ccccc2)C)C)CC1 C#CCC(O)C(=O)NCCC(C)NC(c1c(C)ncn1O)=O C1(CC(=O)N(CC(=O)OCC)CC#C)CN(CC)CC1C(F)(F)F C(=O)(C1=CCCSC1)NC1(C)CCN(C(Cc2c(CC)noc2CC)=O)C1 C1(CC(=O)NCC(N(C(=O)CS(=O)(=O)N(C)C)C)C2CC2)CCCCC1(F)F c1(C(=O)NC2C(C)(CNC(CC=CC)=O)CCC2)cc(NCC)ccc1[N+](=O)[O-] C1(C(=O)NCCC2CCN(C(Cc3c(C)noc3Cl)=O)C2)CC2(CCC2)CO1 Cc1ccc(F)c2c1CN(C(c1cc(F)c(F)c(F)c1)C(=O)NC1CCC1)CC2 N#CC1=C(C(=O)NC2CC(O)CN(C(=O)CCc3c(F)cccc3F)C2)CCC1 C1(CC(N2CC(N(C)C(c3cc(Cl)c[nH]3)=O)C2)=O)CCCCC1O N1(C(C2(COC)CC=CCC2)=O)CCCC(N(C(=O)CNC(N)=O)C)CC1 C1(CNC(c2c(C)noc2C)=O)CCC(C)CN1C(C12COC(CF)(C1)C2)=O c1(C(=O)NCCCN(C(C)C)C(c2ncc(F)cn2)=O)ccc(=O)n2c1CCC2 c1(C(=O)NC(C2CCCN2C(=O)CC(C)CF)C)c(C(F)(F)F)cccc1F c1(CCS(N2CC(O)(C(C)(C)C)C2)(=O)=O)ccc2c(c1)OCCO2 n1(CC(=O)NC2C(C)CN(C(=O)C(C)(C)CF)C2)nc2n(c(=O)c1=O)CCOC2 N1(C(c2c[nH]c(=N)[nH]2)=O)CCC(NC(=O)C2=CCSC2)C(c2ccccc2)CC1 CC(CNC(=O)CNC(C1CC1(Cl)Cl)=O)CN(C)C C(=O)(CC(c1ccccc1)NC(N)=O)NCC(CN(C(=O)COC1CCC1)C)O C(=O)(C(C)(O)C(C)(C)C)NC(CC)CNC(c1csc(C)c1Br)=O c1(OC)ncc(Br)cc1CN1CC2CC2(C(=O)Nc2ccc(O)cc2C)C1 c1(C(CNC(c2cscc2C(F)(F)F)=O)NC(c2cnc[nH]2)=O)ccccc1F C1(C(=O)NCC2CC(NC(c3nn(C)c(O)c3)=O)C2)CCC(C2CCCO2)O1 C1(NC(c2cn(CC)nc2-c2ccccc2)=O)CCCN(C(=O)CN(C)C)CC1 C(=O)(C(F)C(C)CNC(=O)CC1CNC(=O)O1)NC(C=C)CO c1(C(=O)NC(C)CNC(C2(CO)CC2)=O)ccnn1C(C)(C)C O=C(C1=CCCOCC1)NC12CCCN(c3cc(C(F)(F)F)ncn3)CC1C2 c1(C(C2C(NC(c3cscn3)=O)C2)NC(C2(CO)CCC2)=O)ccccc1 C(C(CC(=O)N(C1COC(C)(C)C1)C)NC(C1(c2cc[nH]n2)CC1)=O)OC c1(CC)nc(C)c(C(=O)NCC2(F)CCC(NC(c3cc(Cl)cn3CC)=O)C2)s1 c1(C(C)(C)NC(=O)NC(C(C)N2CCCC2)C2CC2)ccccc1 c1(C(=O)NCCCCCNC(C2(n3cncn3)CC2)=O)sc(Cl)cc1Cl Cc1ccn(CC(=O)N(C(CNC(=O)CCc2cc(C)[nH]n2)C2CC2)C)c(=O)c1 C(=O)(C1=NN2CCC(C)N=C2N1)N1CC(O)(C(C)NC(C(F)=C(C)C)=O)C1 c1(C(N2CCC(NC(C(COC)OC)=O)C(F)C2)=O)ccc2cc(O)ccc2c1 C#CC1CCN(C(=O)CC2CN(C(=O)C3=CCSC3)CC2C)C1 c1(C(N(CCC)CCNC(C2CC(OC)C2)=O)=O)ccc(Cl)c(C)c1O C(=O)(C(CCC(N)=O)N(C)C)NC(C(C)C)C(=O)NC1CCNC(C)CC1 C=CC1(CC(=O)N(CCNC(=O)CN(c2ccncc2)C)C(C)C)CCCCC1 CN1CCC(OCCC(=O)N(C)CC2(NC(C3CCCC(OC)C3)=O)CC2)CC1 C1(NC(=O)Cn2cc(Br)cn2)CN(C(c2ccccc2CO)=O)C2CC12 C1(C(=O)NCC2(C)CSC2)CC2CC1CN(C(=O)CCn1cnc(=N)[nH]1)C2 CCC(CCC(=O)N1CCN(C(C)=O)CC1)NC(=O)CC1CCCOCC1 C1(CNC(c2nc(CC)oc2)=O)C(C)CCN1C(C1CC1(C)CC)=O C(=O)(CCCCC(C)C)NC1C(NC(C(CC(C)C)NC(=O)OC)=O)CC1 CCC(CC)CCC(=O)NC(C)C=CC(N1CCC(CO)C1)=O c1(C(N2CCC(CN(C(C3CCSC(C)C3)=O)CC)CC2)=O)ccc(C)c(C)c1 CC(C)C(C(C)NC(c1ncccc1C1CC1)=O)NC(=O)CCc1ccccc1 CC1(C(=O)N2CCC(C3(NC(=O)CC4=CCC4)CC3)C2)CCCc2ccccc21 C(CCC(C)(C)C(=O)NC1C=CCN(C(=O)CC2(C)CC2)C1)OC CC(C)C(F)C(=O)N1CCSCC1CCNC(C1CCCC(C)C1)=O N1(C(C2C(CC)CCC2)=O)CC(O)(C2CCN(C(c3ncn(CC)n3)=O)CC2)C1 N1(C(CSCCOC)=O)CC(O)CC1C(N1CCCC(NC(C)=O)C1)=O C1(NC(=O)CC2COCC2O)CC12CC(NC(C1CCOCC1)=O)C2 C1(NC(C=C(COC)C)=O)CC2CCC(C1)N2C(C1CC12CCOCC2)=O CC(F)(F)CC(C(=O)N1CC(C)(C#N)C1)NC(=O)OC(C)(C)C C1(NC(C(C)CN(C)C)=O)CC2(CCC(NC(=O)C(F)CC3CCCC3)CC2)C1 Cc1ncncc1C(=O)NC(C)C(C)(C)NC(C1CC(C)(c2ccccc2)C1)=O N1(C(C2(CCC)CC2)=O)CCN(C(c2cc3n(n2)CCC3)=O)CC(C)(F)C1 N1(C(C)=O)CS(=O)(=O)CC1C(=O)NCC(O)CNC(=O)C#CC(C)C c1(CNC(C(C)OC(C)=O)=O)ccc(C(N2CCOCC2CN(C)C)=O)nc1 N1(C(C2N(CC)CCC2)=O)CC(C(=O)NCC=C(C)C)CC(C)C1 C(CCCC(=O)NC1(CN(C)C(c2cnoc2-c2ccc(C)o2)=O)CC1)SC C12(CNC(c3c(C)nc(C(C)C)o3)=O)CCCC1CCN2C(C1CCCCC1)=O N1(C(c2cccc(C(C)C)c2)=O)CC2(C1)CN(C(=O)CC(C)C1CC1)C2 N1(C(C(CC2CN(C(C(CC)OCC)=O)C2)F)=O)CCC(O)(CO)CC1 C1(CNC(CC2(C)CCCO2)=O)COCCN(C(=O)COCC2CC2)C1 CC1(CNC(C2C=CCCN2C(C2CC(C3CC3)C2)=O)=O)CCC(O)CC1 N1(C(c2ccn(C3CC3)n2)=O)CCC2CC2(C(=O)Nc2ccsc2)CC1 C1(C)(CNC(C(F)OC)=O)CCCN(C(c2nccc(C)n2)=O)C1 C(=O)(C(F)(F)C1=CCOCC1)N1CC(CNC(C(C(C)C)O)=O)C2(C1)CC2 NS(=O)(=O)CCCN(C(=O)NC1CC1c1cn[nH]c1)Cc1ccc(O)cc1 Cn1nc(C(=O)NC(CO)CCCNC(C2CCCSC2)=O)cc1F C1(C(=O)NCC2CCC(CN(C)C(C3CC34CC4)=O)CC2)CCC2(CCC2)O1 C1(N(C(COCC(C)C)=O)C)CCN(C(c2n[nH]c3c2CCC3)=O)CC12CC2 C(C(C)(O)C(C)C)NC(C1C(CNC(COC)=O)CCC1)=O N1(C(=O)C(C2CC(F)(F)C2)O)CCCC12CCS(=O)(=O)CC2 C12(NC(c3c(C)n[nH]c3)=O)CC3CCC(C1C2)N3C(C12CCCCN1CCC2)=O C1(NC(=O)CCc2cc(Br)cs2)CN(C(c2cnsc2)=O)CC1O N1(C(COCCC)=O)CCCC(O)(CNC(=O)COC2CCCCCC2)C1 C(=O)(CCCCCCc1c[nH]c2ccccc12)NCC1(OC)COC1 CC1(NC(C2CC2(Cl)Cl)=O)CCN(C(C2(Cc3cccs3)CC2)=O)C1 c1(C(=O)NCc2scc(CNC(C(CSC)O)=O)n2)ccnc(C)c1 NC(=O)CCCCC(=O)N1CC(C(=O)NC2CCC3(CC2)CC3)C(F)C1 N1(C(C2C(C)OC(C)C2C)=O)CC2(COC(CNC(C3CCC(F)(F)C3)=O)C2)C1 C(C)(C(C(=O)N1CCCCC1C(=O)NCc1nc(C)c(C)[nH]1)N(C)C)OC N1(C(C(=O)NCC)=O)CCCC12CCN(C(=O)CC1CCCO1)CC2 C1(C(NOCCN(C)C)=O)CCC(C2CC2)N1C(=O)C=Cc1ccncn1 Cc1ccc(C)c(CC(=O)NC(C2CCCN2C(=O)Cc2coc(C)n2)(C)C)c1 C(=O)(C1=C(C#N)CCC1)NC(C1CCCCC1)C(=O)NCC(C(C)(C)O)F C1(N(C)C)CN(C(C2(C3CCCO3)CC2)=O)CC1CO.c12cnccc1NC2=O C(CC(O)C(=O)NCCC(=O)NC(c1csc(C)n1)C)SC C(=O)(CC(C)(C)CNC(=O)C=Cc1ccnn1C)N1C(CC)CCCC1 C1(C(=O)NC(C)C)CCCC12CCN(C(c1cc(F)c[nH]1)=O)C2 c1(C(N2C(C(N(CC)Cc3ccoc3CC)=O)CCC2)=O)ncncc1C N1(C(c2cc(C(C)=O)on2)=O)CC2(NC(C3CC(F)(F)C3)=O)CC1C2 c1(-n2cc(C(N(C(c3n(CC)nc(C)c3)=O)C)C)nn2)cc(F)cc(Br)c1 c1(C(=O)NC(CNC(c2cccc(CC)c2)=O)C(C)C)nc(C)ccc1Br C1(CCC)(NC(c2c[nH]nc2OC)=O)CCCN(C(c2cncc(SC)c2)=O)C1 N1(C(Cn2ccc(C)n2)=O)CCC(NC(c2cc(C(F)F)ccc2F)=O)C(F)C1 C(=O)(N=c1cc[nH]cc1C1CC1)Nc1c(C)ncc(Cl)c1 c1(OC)ccc2nccc(CNC(=O)NCC(C)(O)C3CC3)c2c1 C=C(C)CC(C(=O)NC1CC(OCC(=O)NCCC#CCC)C1)OC Cc1c(CCNC(C2CC(C)N(C(=O)C=CC(C)(C)C)C2)=O)cnn1C CC(C)CCC(F)C(=O)NC(C)(C)C=CC(=O)NCC1COCC(=O)N1C C(=O)(C1NCc2nc(C)ncc21)N1CC(C2OCC(C(=O)OC)C2)C1.C1CS1 C(=O)(C1=NNC(=O)C1)N1C(CN(C(C(CCC)N(C)C)=O)C2CC2)CCC1 C1(c2nc(CNC(C=C(COC)C)=O)[nH]n2)CCN(C(C23CC(C)C2C3)=O)CC1 c1(C(=O)NCC(C(C)(C)C)NC(C2N(CCC)C(=O)CC2)=O)cc(F)ccc1C C(C(C)(CO)NC(c1cn(C(F)(F)CO)nn1)=O)NC(C(C)NC(=O)NC)=O N1(C(C(C2CN(C(C=CC(C)C)=O)C2)O)=O)CCC2(CC=CCO2)C1 C1(NC(C(C(C)C)O)=O)CN(C(c2cnc(C(F)(F)F)s2)=O)C2(CCOCC2)C1 C(=O)(CS(=O)(=O)C1CC1)NC1C(CNC(C2C(C)=C2)=O)CCCC1 C12(NC(c3cnc(C)o3)=O)CCCC1CN(C(=O)Cn1cc(C3CCC3)nn1)C2 c1(NC(C)=O)cc(CN2CC3CC3(C(=O)NC(C)C3CC3)C2)ccn1 n1(CC)nc(CS(=O)(=O)Nc2ccccc2NC(=O)OC(C)(C)C)c(C)n1 N1(C(CC(C=C)C)=O)CCC2(CC1)CCN(C(C)=O)CC2C Cc1cc(N)cnc1C(=O)NC1CC(CCNC(=O)CC2CCC(F)(F)CO2)C1 Cc1nc(C2CC2)oc1C(=O)N(C(C)CCNC(=O)Cc1ccoc1Cl)C c1(C(=O)NCC(C)(C2CCC2)NC(c2cnc(S)[nH]2)=O)csc(C(F)(F)F)n1 Cn1ncnc1CCC(=O)NCCN(C(=O)CCCC1CCCC1)C1CC1 C(C(CN=C(NC(C)CSC)NC1CCC2(C1)OCCO2)C(C)C)OCC.C(C)(C)O N1(C(C=C(C)CNC(c2scc(C)c2C)=O)=O)CCN(C)CC(C)C1 c1(C(N(CC(C)CNC(C2CC3CCC(C2)S3)=O)C)=O)coc(S(C)(=O)=O)c1 c1(NC(C(CCOC)NC(c2ccnnc2)=O)=O)cnc(C)c(C#N)c1 N1(C(CC2CCC(C)(C)C2)=O)CCCCC(C(=O)NCC2CC3(C2)CC(O)C3)C1 C1(CNC(CCC(=C)Cl)=O)C(C2CC2)CCN1C(=O)C=Cc1c[nH]c(=N)c(C)c1 CC(O)(CNC(c1sccc1C1CC1)=O)CNC(C1CC1c1ccccc1)=O Cc1ccc2c(c1)CC(C(=O)NC(C)(C)CNC(=O)CC1CCC3(CC1)CC3)S2 C(CCN=c1ccc(C(F)(F)C(F)(F)F)n[nH]1)NC(c1c(C)nccc1)=O N1(C(c2c(C)ccnc2)=O)CCC(C2(NC(C3CCC(CCO)CC3)=O)CC2)C1 CCCCC(O)C(=O)NC1CCN(C(c2cn(C(C)COC)nc2C)=O)C1(C)C CN1CCC(C(=O)N(C)CCNC(=O)CCc2cncn2C)CC1 N1(Cc2ccc(NC(C)=O)s2)CCCC(C)(C(=O)NCC2CS(=O)(=O)CCO2)C1 CC1(C)CC(C(N2CC(F)(CO)C2)=O)N(C(c2cnc3n2CCC3)=O)C1 C(C(COC)CC(=O)N1CC(C(=O)N(CC(C)OC)C)C(C)C1)OC N1(C(C(C)OCCC=C)=O)CCN(C(=O)C=Cc2ccc(Cl)cc2)C2(CC2)C1 C(CC)(C(=O)NCC#CC(=O)N1CCCC1C1(C)CC1)OCC CCCCC(CNC(=O)C=C(Cl)Cl)NC(=O)C(O)COCc1ccccc1 c1(C(N(CC(C)C(=O)NCCCCC2CC2C)C)=O)ccc(O)nc1 c1(OC)cncc(C=CC(=O)N(CC(C)N(C(=O)CCCn2ccnc2)C)C)c1 N1(C(c2cc(Cl)n[nH]2)=O)CCCc2cc(-c3ccccc3F)ccc21 CCC(CC(C)C)C(=O)NCC1(CNC(=O)C(C)CC2CCCC2)CCC1 c1(C(N(C(CN(C(c2c(C)ccnc2)=O)C)C)C)=O)[nH]ccc(=O)c1C Cn1nnc(C(=O)NCC(CO)NC(c2ccc(O)nc2)=O)c1N CC(C)(C)C(=O)C(=O)N1CC=CC(C(=O)NOCCC2CC2)C1 C=C(Cl)C(C)(C)C(=O)N1CCC(O)(CNC(C2CCCC(=O)N2)=O)C1 C1(COC)(NC(c2c(Cl)ccnc2C)=O)CCCN(C(c2cccc(N)c2)=O)C1 C1(NC(c2c(CC)ncs2)=O)CCOCC1NC(=O)CSc1nnnn1C1CC1 C1(CNC(c2c(CC)c[nH]c2)=O)CC(NC(=O)CCCc2cnccn2)C(O)C1 N1(C(c2sc(Br)cc2Cl)=O)CCCC2CNCCCC12 c1(C(=O)NCC2CN(C(c3cnn(CC)n3)=O)C2)c(Br)nc2n1CCC2 C1(OC)CN(C(=O)C(C)C(F)F)CC1NC(c1cc(C2CCCCC2)[nH]n1)=O C(=O)(C(C)(C)C(=O)NC(CNC(c1ccccc1OC1CC1)=O)C1CCC1)NC C1(C(=O)OC)CCC(n2nnnc2C(C)NCCn2cc(NS(C)(=O)=O)nn2)C1 CCC(CC(=O)N1CCC(CC)C1CNC(c1cnncc1O)=O)C1CCC1 Cc1cccc(F)c1NC(=O)CN(C(=O)CN1C(C)CCC1C)CC1CC1 n1(CC(=O)NCC(C2CCC2)NC(c2ncn(C)c2)=O)ncccc1=O c1(OC)ccc(C)c(C(=O)N(C)CC2CCN(C(=O)C(C)S(C)(=O)=O)C2)c1N C1(C(N(CC(C)(C)C)C)=O)CN(C(=O)CN2CCSCC2)CC12CC2 c1(CC)cc(C(N2CCSCC2C(=O)NC2(CCO)CCC2)=O)c(C)o1 C1(C(=O)NC2(C3CN(C(C4N(C(N)=O)CCC4)=O)C3)CC2)CCn2cncc2C1 C1(C(=O)NC23CC(F)(C2)C3)(CC)CCN(C(=O)C2=CCCC2)CC1 C1(NC(C(=O)NCC(CNC(C(CC=CC)C)=O)OC)=O)CCC(F)(F)CC1 c1(C(=O)OC)cc(Cl)c(N2CCC(CCNC(c3[nH]c(C)nc3C)=O)C2)nc1C C#CCCCCC(=O)N1CC2(C)CC1(C(=O)NCCOC1CCOC1)C2 c1(N2CCN(CC#CC)CC2)ncnc(C)c1C#N C1(CC(=O)NCC2CC(NC(c3ccc([N+](=O)[O-])o3)=O)C2)CC(=O)NC(=O)C1 Cc1nncc(C(N2CCC2CC(N2CCC3(CCC3)C2)=O)=O)c1C c1(C(=O)NCCSCC(=O)NC(C(CCC)O)CO)ccc(C#N)cc1C C1(NC(C2(C#C)CCC2)=O)CN(C(c2c(C)nn(C)c2Cl)=O)CCC1C N1(C(C2N(C(C(C)Cc3ccccc3)=O)C3CCC2C3)=O)CCCC(C)(O)CC1 c1(CNC(C2C(OCC)C2)=O)ccc(C#N)c(C2CC2)n1 N1(C(CC(CC)C)=O)CCCCC(CCC(=O)NCCc2ccc(F)cc2)C1 c1(OC)cccc(C(=O)NCC(CO)NC(=O)CCc2ncccc2C)c1 N1(C(C(=O)NCc2ccccc2)=O)CCCC2(NC(=O)C=CCl)CC12.CC(F)(F)F c1(C(=O)NC(CNC(C2(CCC=C)CC2)=O)CCC)onc2c1CCCC2 C1(CNC(=O)Cn2cc(Cl)cn2)C2CN(C(c3cnncc3O)=O)CC12 C#CCCCC(=O)NCC(c1ccc(C)cc1)NC(C1(C)COC(=O)N1)=O c1(C2C(C(N(CC(CC)NC(=O)C=Cc3cnc[nH]3)C)=O)C2)cccc(Cl)c1 Cc1cc(O)c(Cl)cc1C(=O)NC1(CCCNC(C2C=CCCC2)=O)CC1 C(c1cccnc1)=CC(=O)NCCC1N(C(C(CC)F)=O)CCC1 CC1(CCNC(C2(C)COCCO2)=O)CCN(C(c2ccccc2C2CC2)=O)C1 C1(NC(c2ccc[n+]([O-])c2)=O)CC(O)CN(C(=O)CCC=CBr)C1 c1(CNC(CN(CCC)C(C2CCC(=O)N2)=O)=O)cccnc1OC c1(N)c(N(C)C)cccc1NC(c1ccccc1SC)c1n(CC=C)nnn1 Cc1cccc(C(=O)N(Cc2nc(C(C)C)no2)CC2CC(Cl)=NO2)c1 N1(C(C2CC23CC3(F)F)=O)CC2(CCN2C(C2CCCC2)=O)C1 C1(C)(CC)CC(C(=O)NCC(C2CCNCC2)C)CCO1 C1(C(=O)NC2C3CCN(C(=O)OC(C)(C)C)C32)CC2CCCC(O)(C1)C2 N1(C(c2c(OCC)cccc2)=O)CCCCC(NC(=O)C=C2CCSCC2)CC1 N1(C(c2n(CCCC)ncc2)=O)CC(C)C(C)(CNC(=O)CCOCC(C)C)C1 C1(CC=C)(C(=O)NCC2(O)CSC2)CCCN1C(=O)CCC1CCCN1C N1(C(CCSCCN(C)C)=O)CC2(CC(NC(c3cnc(C(F)(F)F)s3)=O)C2)C1 C1(NC(Cc2cccc(OC)n2)=O)CCN(c2ccnc(C)n2)CCC1CO Cc1cc(N)cnc1C(=O)NC(C(=O)N(C1CC2CC2C1)C)c1ccoc1 N1(C(c2cc(C)c(Cl)s2)=O)CCN(C(c2cscc2Cl)=O)CC1C C1(NC(C2(CCC=C)CCCC2)=O)CCCCC1CNC(=O)C1=CSCS1 N1(C(CCCNC(=O)OCC)=O)CCCN(C(=O)CC2(CO)CCCC2)CC1C C1(C(N(C2CCCN(C(c3ccc(CO)s3)=O)C2)CC)=O)C(C)(C)C1(C)C c1(CC(=O)NCC23CC(NC(C(C)OC(C)(C)C)=O)(C2)C3)cnn2ccccc12 Cc1cc2[nH]c(C(=O)NC3CCN(C(=O)C(C)(C)CC#N)CC3C)cc2o1 N1(CC(=O)Nc2ncc(C(=O)OCC)s2)CCC(O)(CO)C1 C1(C(N(CCCNC(=O)C(C)Cc2ccco2)C(C)C)=O)CCc2ncnn2C1 c1(C(N(CC(CN(C(c2c(C)c[nH]n2)=O)C)O)C)=O)coc2c(C)cccc12 O=C(CCN=C(NCc1cccs1)N1CCC(NCC2CC2)C1)N1CC1 N1(C(CS(CCCC)(=O)=O)=O)CC2CCCC2(N=c2nc(C3CC3)[nH]s2)C1 CC1CN(C(=O)CC2CC(=O)NC2=O)CC(C)CN1C(=O)C=CBr c1(N2CCCC(NC(C3CCC(C)(CC)O3)=O)C2)nc2cccnc2s1 N1(C(CC2CN(C)C2)=O)CCCC1CCNC(=O)Cn1cnnn1 c1(OCCC(=O)NC(CNC(C2(n3ccnn3)CC2)=O)CO)cccc(Cl)c1Cl C1(OC)(CNC(=O)CC(=O)NCC(F)(F)F)CCN(C(=O)CC2(C)CC2)C1 c1(C(N(CCCCN(C)C(C2CCC(O)C2)=O)C)=O)[nH]nnc1-c1ccccc1 C=CCC(C)(CC)C(=O)N1CCCC(NC(c2c(C)cc(OC)cc2F)=O)CC1 N1(C(C(C(C)C)O)=O)CCC(NC(=O)C=CCF)C(O)C1 c1(C(=O)NC2CCC(NC(C(N(C)C)C3CC3)=O)CC2)c[nH]c2ccc(F)cc12 c1(NC(C(c2cnc(C3CC3)s2)N(C(CC#C)C)C)=O)ccc(Cl)cc1 CC(C)(CNC(c1cccc(-c2ccoc2)c1)=O)CCNC(=O)CNC(N)=O C(=O)(CN=c1cc[nH]cc1)N(CCN(C(=O)C(CO)C(C)(C)C)C(C)C)C c1(C(C)C(=O)NC2(CNC(=O)C(CC3CC3)N(C)C)CC2)ccc(F)cc1F CC1OCCN(C(c2cn(C)nn2)=O)C1C(=O)NCC1CC1C1CCC1 CCC(CN=c1nc(N(C)CCc2ccccc2F)c2sccc2[nH]1)C(C)(F)F c1(CCCC)n[nH]c(=NC(=O)NC2CCC(O)CC2)s1 c1(NC(C(CCSC)O)=O)ccc(NC(C2CN(C(C)=O)C2)=O)c(C)c1 C1(NC(C(C)NC(=O)NC)=O)CCSC12CN(C(c1scnc1C(C)(C)C)=O)C2 N1(C(CSCC#C)=O)CCC(N=c2[nH]nc(C(=O)OC)o2)C(CC)C1 c1(CC)cc(CN(C)C(=O)NCc2csc(C(F)F)n2)cc(OC)c1OC c1(CCC(=O)NCC(C)NC(C2CC2c2ccsc2)=O)cccc2c1OCO2 CCCCCCC(C)C(=O)N1CCC(CCC(=O)NCC(C)C#N)CC1 C1(C(CNC)=O)CCC(C(=O)NC(CCO)CC(C)C)(OC)CC1 CCC(C)CC(C(=O)N(C)Cc1ccc(C)cc1)NC(c1cc(C#N)c[nH]1)=O c1(C(CNC(c2c(CC)nco2)=O)NC(=O)CCSC)ccccc1OC C1(C(=O)OC)Cc2c(C)cccc2CN1C(=O)C(=O)Nc1cccnc1 C1(NC(COCP(C)(C)=O)=O)CN(C(=O)CN2CCSCC2)C2(CCOC2)C1 C1(C(N2C(C(C)NC(CCC(=C)Br)=O)CCC2)=O)COC(C)(C)CO1 N1(C(C2C(CC)N(C)CC2)=O)CCC2CN(C(c3ncc(Br)cc3C)=O)C2C1 c1(C(=O)NC2C(C)CCN(CCC3CC3)C2)cc2ccccc2s1 N1(C(CNS(C)(=O)=O)=O)CC2CC(C1)CN(C(=O)C=Cc1ccco1)C2 CC1CN(C(=O)CC(C)n2cccn2)CC1CNC(=O)C(F)=CC1CC1 C1(CNC(=O)C=CCn2cncn2)CC(F)(F)CN1C(c1cccc(CF)c1)=O N1(C(C2CN(C(Cc3c(C)noc3C)=O)CC(C)C2)=O)CCc2ccccc2C1 CC1OC2(C)CC1(C(N1CC3CC3(NC(=O)CC3CCCCC3O)C1)=O)C2 CCC(CC)(CC)C(=O)N1CCCC(NC(C2CCCN(C(C)C)C2)=O)CC1 C(=O)(N1CC(C)(O)CO1)C1CCN(C(c2cc(CC)[nH]n2)=O)C1CC C1(C(=O)Nc2cc(Br)cc(Cl)n2)CN(C(c2ccc(O)cn2)=O)CC(F)(F)C1 S(=O)(=O)(C1CCOCC1)NCC1N(C(C(C(C)C)O)=O)CCCC1 c1(C(=O)NC(CC=C)CNC(=O)Cc2csc(S)n2)cnc2c(cnn2C)c1N N1(C(C(C2(O)CN(C(c3nn(C)c(F)c3)=O)C2)F)=O)CCC2(CSC2)C1 C1(C(=O)NCC#CC(=O)NCC(C)C2CC2)C2CC3C(C2=O)C13 c1(C(=O)NC(C2CCN(C(C3(C)CCCN3C)=O)C2)C)nc2ncccn2n1 N1(C(CC(CC)OC)=O)CC2CC(C1)C2NC(c1ccc(C(F)F)s1)=O N1(C(CC(N2CCC(C)C2)=O)=O)CCOC(CC(c2ccccc2)O)C1 N(C(=NCCN1CCCC1)NC1CCCC(C)(C)C1)CCOC(C)(C)C N1(C(C2C(CCC)C2)=O)CC2CCC1CN2C(C1(OC)CCSC1)=O C1(C(=O)NC2CN(C(c3n(CC)ncc3)=O)CC23CC3)CCc2c(nnn2C)C1 C#CCC(O)C(=O)N1CC(C(=O)N(C)CC2COC(=O)N2)(SC)C1 c1(CCNC(CN(C)C(N)=O)=O)ocnc1CNC(=O)CCc1cnn[nH]1 c1(C(N2CC(NC(C(C)P(C)(C)=O)=O)C(O)CC2)=O)ccc2n[nH]cc2c1 C#CCC(C)(C)C(=O)NCCCNC(=O)C(C)Cc1ccc(Cl)c(Cl)c1 C(CCCC(C)(C)NC(=O)Cc1ncn2c1CCC2)NC(C1C(CC)CCC1)=O C(=O)(C(C)(C)CC(=O)N1CCC(O)(CCNC(=O)CN2CCCNC2=O)C1)OC N1(CC)CCCC1CC(=O)NCC(CCOC)NC(C1(C)CC1C)=O Cc1cc(C(=O)NCCC(C)NC(=O)Cc2cncs2)ncc1C#N C1(CC(=O)NCC(CN(C(C2COC(=O)C2)=O)CC)(C)C)CCN(C(C)=O)CC1 C1(CCCCNC(c2ccc(C(F)F)nc2)=O)CCCN(C(=O)C(F)(F)CO)C1 N1(C(C(=O)N(C)C)=O)CCCC2(CNC(c3nc[nH]c4nccc3-4)=O)CCCC12 c1(SCC(=O)NCC2CN(C(C(C(C)C)O)=O)CC(F)C2)ccc([N+](=O)[O-])cc1 CC1C(NC(c2cc(-c3ccco3)on2)=O)CCCN1C(C1CS(=O)(=O)C1)=O C1(CNC(c2onc(CC)c2C)=O)CN(C(C2CC3CCC2O3)=O)CCCO1 c1(CN=C(NC2CCN(C(CCC=C)=O)C2)NC(C)C)cc(C)nc(O)c1 CC1=C(C(=O)NCC2(F)CCN(C(c3c[nH]c(=N)s3)=O)C2)CC1 C1(NC(C2CN(CC)C2)=O)CCN(C)CC1OC.c1(C(C(=O)OC)C)ccccn1 c1(C(C)OC)ccc(S(=O)(=O)NC)s1.c12cc(F)cc(c1C)NC2=O N1(C(C(c2c(C)cccc2)(C)C)=O)CC2CC1CC2CNC(=O)C(C)NC(N)=O C1(NC(c2cc(C)on2)=O)CCCC12CCN(C(c1cccc(N(C)C)n1)=O)C2 C1(NC(CC(CC)OC)=O)CCC2CC1CN2C(C1(C#N)CCOC1)=O c1(NC(CC(=O)OCC)C)nc2cccc(C#N)c2n1C N1(C(C=NOC)=O)CC2CCN(C(c3cc4scnc4[nH]3)=O)CC12 CC(CC(N)=O)C(=O)NCC1CCN1C(c1cc(-c2ccc(O)cc2)on1)=O C1(C(NOCC(=O)NCC2(C)COC2)=O)CCC(F)C1 C1(CCNC(c2c(C)nc(CO)s2)=O)CN(C(=O)CNC=O)CCS1(=O)=O N1(C(C)=O)CCOCC1C(N1CCC(C)(CCNC(=O)C2=CCC2)C1)=O C1(CNC(C2(N(C)C)CC2)=O)CC(C(C)(C)C)CCN1C(c1coc(Cl)n1)=O C(=O)(CS(=O)(=O)CCO)N1CC(OCCNC(c2ccc(N)cc2F)=O)C1 C12CC3CN(CC13)C2=O.C1(CNCC)CCCN(c2cc(OC)ncn2)C1 c1(C(N(C(C)C)C)=O)n[nH]c2c1CCN(Cc1cc3c(cc1Br)OCO3)C2 Cc1nc(C)c(C(N2CCC(NC(=O)CC3CCCC(C)C3)C2)=O)c(C)n1 c1(C(N2C(CCNC(CC3CC(C)(C)C3)=O)COCC2)=O)ccc2cc[nH]c2c1 Cc1cc(C(=O)NC(C2(O)CCN(C(C3(N(C)C)CCC3)=O)C2)C)cnc1O c1(CC)occ(C)c1C(=O)NCCCN(CCCNC(=O)CN1CCSCC1)C C12(NC(CN(C)CC)=O)CCC(CNC(C3C4CCCCCCC34)=O)(CC1)OC2 N1(C(=O)OC(C)(C)C)CC(C(=O)NCC#CCNC(=O)Cc2ccsn2)C1 c1(C(=O)NC(C(C)NC(=O)C=CCO)(C)C)ccc(S2(=O)=NCCC2)cc1 Cc1cc(C(N2CCC(NC(=O)C(C)(Cl)Cl)C(CO)C2)=O)cc(N)c1Cl C1(CNC(=O)C(F)C2CCC2)CCCN1CC(=O)N(c1ccccc1)C1CC1 O=C1CC(C(=O)NCCC2CCN(C(c3ccn(CCF)n3)=O)C2)(CF)C1 c1(OC)cccc2c1OCCCC2NC(=O)C(=O)NC(CO)C(C)C c1(NC(=O)NCC)ccc(C)cc1C(=O)NCC12CC(CN1C)C2 c1(C(N(C2CC23CC3)C2CC2)=O)nc(Br)cnc1N.CCC(CNC=O)N c1(C(=O)NC2CC(SC)C2)cc(C#N)ccc1O.c12cn(C)c(n1)C(=O)N2 c1(C(=O)NCC2(CCNC(=O)CC3(O)CC3)CC2)csc(C(F)(F)F)c1 N1(CC(Cc2cn(C(COCC)C(=O)OC)nn2)O)Cc2ccccc2C1 C1(CC(N2CC(C(N)=O)C2)=O)C2CCCC2N1C(C1(O)CCCCC1)=O c1(C(N2CCC(CC=C)(NC(c3cn(C)cc3C)=O)C2)=O)cccc2ccsc12 c1(C(N(C2CC3(CCNCC3)C2)C2CC(C)C2)=O)cc2cc(Br)ccn2n1 N1(C(Cc2scc(C)n2)=O)CC2(C1)CN(C(c1ccnc(C3CC3)n1)=O)C2 C1(NC(C2CCCN(CC)C2)=O)CCN(C(C2CCS(=O)(=O)C2)=O)CCC1CO c1(C(=O)NC2C(C)N(C(c3cnnc(O)c3)=O)CC2)ccc2c(c1)CCOC2 N1(C(CCc2ccc(OC)cc2)=O)CCC(F)(C(=O)Nc2ccc(Br)nc2)CC1 C1(CN(C(C=CC)=O)CC)CCCN(C(=O)C(C)CCC)C1 C1(SCC)CCC(C(=O)NCC2(CNC(C3COC(=O)N3)=O)CCC2)CC1 CN1N=C(C(=O)NC2(CNC(=O)CC3CC(F)(F)C3)CCCC2)CCC1=O c1(C(=O)OC)cc2[nH]ccc2cc1NC(=O)Cc1cccc(C(C)C)c1 c1(OC)csc(C(=O)NC(CNC(C2COCC2(C)C)=O)C(C)C)c1OC C1(C(=O)NC(CCCC)CNC(=O)CCC(=O)NC2CCCC2)CCCS(=O)(=O)C1 C1(CS(=O)(=O)NCC2CC(C)OC2)CC(C)(C)OC1(C)C Cc1cnc(C(=O)NC2CCC(N(C(=O)C(C)n3cccn3)C)CC2)c(F)c1 c1(C(C(=O)NC2CC(F)(CNC(COC)=O)C2)O)cccc([N+](=O)[O-])c1 Cc1cc(C#N)ccc1C(=O)NC(C)C(C)C(=O)NCC1CN(C)CCN1C C1(CNC(=O)Cc2csnn2)CC2CCC1N2C(C1CCC2CC2C1)=O c1(C(=O)NCC(CO)NC(c2[nH]n(C)c(=O)n2)=O)c[nH]c2cccnc12 N1(C(C2C(C=C)CC2)=O)CC(NC(c2snnc2C(C)C)=O)CC(C)(C)C1 CCCC(C)(O)C(=O)N1CCC(CC(N2CC3CCC3(OC)C2)=O)CC1 C(=O)(C#CC1CCC1)N(C1CCC(NC(CN(C2CCCC2)C)=O)C1)C c1(C(=O)NCC(CNC(=O)CCCCCF)CO)ccc2nc[nH]c2n1 c1(N(CC)CC)ccc(S(=O)(=O)N2CCc3cc(OC)ccc32)c2ccncc12 N1(C(C(CC=C)(C)C)=O)CCC(C2CC2)(CNC(C2(OC)CCOCC2)=O)C1 C1(O)(CCNC(c2nc(C)sc2)=O)CCN(C(=O)Cc2ccc(O)cn2)C1 c1(OC)c(O)cc(C(=O)NC(c2ccc(O)nc2)C)cc1C#N C(N=c1[nH]cnc(NCC(C)Cn2nc(C)cc2C)c1C)c1occ(C)c1 Cc1cc(F)cc(C(N2CCN(Cc3c(F)cc(O)cc3F)C3CC23)=O)c1O C(=O)(C#CC1CCCO1)NCC1CC(NC(C(C(C)C)O)=O)C1 c1(C(C(=O)NCC2(F)CC(CNC(C3CC(=C)C3)=O)C2)O)ccccc1Cl N1(C(C2(C)CCC2)=O)CCC2CN(C(=O)CON=C3CCCCCC3)CC2CC1 c1(C(N2CCC(OCCCC(=O)OC)CC2)=O)cc(Br)c(C)cc1Br C1(CNC(=O)CC2CCC3CC23)CCCN(C(c2cc(=O)cc[nH]2)=O)C1 Cc1cccc(C(=O)NC2CC2CNC(c2ccc(NC(N)=O)cc2)=O)c1C CC(C)CCCCCC(=O)N1CCN(C(=O)C(C)(C)CC2CC2)CC1CO c1(C(=O)NCC2(C)CCC(NC(c3ncn(C)c3)=O)C2)nc2cnccc2s1 N1(C(COCC#C)=O)CC(CNC(=O)Cc2c(C)nc(O)nc2C)C2(CCC2)C1 C=C(F)C1(CC(N2CCCC2C2(C(=O)NC3CC(=O)N(O)C3)CC2)=O)CCC1 C(C(C)(C)CC(=O)N1CCC(CO)C1)NC(C1(C#N)C(C)C1)=O c1(CC(N2C(C(C)NC(C3CC3OCF)=O)CCC2)=O)ccc(OC(F)F)cc1 N1(C(c2c(CC)cncc2)=O)CC2C=CC1C(C(=O)NCC(C)(COC)CC)C2 c1(C(=O)NC(CC(C)NC(=O)CCc2nccs2)C)nccnc1O N1(C(C(C)(CO)OC)=O)CCN(C(c2cc3ccccc3cn2)=O)CC12CCC2 c1(C(=O)NC2C(CNC(CCCC(N)=O)=O)C2)cc2cc(Br)cnc2s1 CC(CNC(C1CC1C(N)=O)=O)(CO)NC(=O)CC=CCc1ccccc1 c1(CCNC(=O)Nc2nc(C(=O)OCC)c(CC)s2)ccc(F)c(F)c1 C(CN=c1nc2c(cnn2C)c(NCCc2n[nH]c(O)n2)[nH]1)N(CCOC)C CC1(C(N2CCCCC2CNC(C2CCCC2CF)=O)=O)CCOCC1 c1(C(N2CC3C(C(=O)Nc4cnc(OC)nc4)(C3)C2)=O)ccc(C)nc1Br Cc1cc(C(=O)N(CC(O)CNC(c2cc(CO)n(C)n2)=O)C)[nH]c1C C1(C#C)(NC(C2(CC#C)CN(C(c3coc(C)c3)=O)C2)=O)CC2CCCC12 N1(C(C(COC)CC(C)C)=O)CCCC2C(NC(c3cc(Cl)ns3)=O)C(C)(C)C12 CC1=NC(Cl)(C(F)(F)F)C(N2CCC(CCNC(C3(CC4CC4)CC3)=O)C2)=N1 C(C(C)N=c1[nH]c2ncnc-2c(-c2ccccc2)[nH]1)NC(c1ccnc(C)n1)=O N1(C(C(c2ccc(F)cc2)C)=O)CC(NC(C2CCC(=O)C2)=O)C(C)C1 Cc1cccc(CNC(=O)OC2CC2(F)F)c1.C12(O)CN(C1)C(=O)CCNC2=O c1(C(N(CCCNC(C2COCC2C(N)=O)=O)CC)=O)cc(C)cc(Cl)c1 N1(C(c2c(C)cn(C)c2)=O)CCC(F)CC1C(=O)NCC1CCCN1C C12(C(=O)NCCC3C(C)CCCN3C(C34CC(C3)C4)=O)CCC(CC1)C2(C)C N1(C(c2ccn(C)n2)=O)C(CNC(c2[nH]nnc2C2CC2)=O)CC2CC12 C1(F)(CNC(CCNC(COC)=O)=O)CN(C(=O)CC2CCC(C)O2)C1 c1(C(N(CCCOCCN(C(c2c(C)cc[nH]2)=O)C)C)=O)c(C)noc1C(C)C N1(C(C23N(C(C(CC(C)C)OC)=O)CC(C)(C2)C3)=O)CCC2CCCC2C1 C1(NC(C(c2cc(C)sc2)(C)C)=O)COCCN(C(C23CCCC2CCC3)=O)C1 N1(C(=O)OC(C)(C)C)C2CCC(NC(C3(F)CCN(C(C)=O)C3)=O)C1CC2 C1(CNC(C23CCN(CC2)CC3)=O)CC12CCN(C(C13CSC(C1)C3)=O)CC2 C(=O)(C(C)C(O)C(C)C)N1CCC(C(=O)N(C2CCN(OC)CC2)C)(OC)C1 C(=O)(C#CC(C)(C)C)N(C)Cc1cn(CC2CC3CC3C2)nn1 c1(CC)cc(C(=O)N(CCCNC(c2cncc(O)c2)=O)C)cc(Cl)n1 C1(NC(CN2CC(CC)C2)=O)CCN(C(=O)C(c2ccccc2Cl)C)CC1C Cc1nc(CC(=O)NC(c2cn(C)nn2)C(NCP(C)(C)=O)=O)n[nH]1 N1(c2ncc(C#C)cn2)CCCC12CCN(C(=O)Cn1ccsc1=N)CC2 c1(C(=O)NCCN(C(C2(CC=C)CC2)=O)C)cnn(C)c1CC C(=O)(CCCCCC(C)(C)C)NCCC1CCN(C(C2CC(C)=C(C)CC2)=O)C1 C1(NC(C(C)SC)=O)CC2CCC(C1C)N2C(=O)CCCCCF c1(C(=O)NC(C)CCCNC(C2(C#N)CC=CC2)=O)cnc2c(c1)CCCC2 N1(C(CC#N)=O)CCCC(C(C)NC(C2CC(=O)NC2=O)=O)C1 c1(C(=O)NC(CCCNC(C=CC(CC)C)=O)C)nccnc1C C1(CNC(c2cc(CC)ncn2)=O)CN(C(c2nccn2C(C)C)=O)CCN1C C1(C(=O)Nc2c(OC)ccnc2)CCC2(CC2)N1C(c1c[nH]nc1Cl)=O c1(C(=O)NCC(CCCC)NC(=O)CC2CN(C)C2)nc2ncccn2n1 Cc1c(C(=O)NCC2C(C)CCCN2C(=O)CCCc2ccsc2)c(Cl)nn1C C(C(=O)N=c1cc(C(F)F)[nH][nH]1)c1ccc(OC)nc1 C(CNC(C1C(C)C1C)=O)(CC(C)C)NC(CC(=O)NCC)=O c1(C(N(C)CC2CN(C(c3cncn3C)=O)C2)=O)cccc(=O)n1C N1(C(c2nc(C)oc2C)=O)CC(C(=O)NC2(C)CC3CCC2C3)C2(CCC2)C1 CC1CCC=C1C(=O)N1C2CCC1C(CNC(=O)CN1CC(=O)NC1=O)C2 N1(C(CC(=O)NCC#C)=O)C2CCCC1CN(C(C1(C)CCCC1(F)F)=O)C2 C1(C2CCSCC2)(C(=O)NCCCC2CCN(C3C(C(C)(C)C)CCC3)C2)CC1 Cc1sc(NC(=O)CN2CCSC(C(C)C)C2)c(C)c1C C1(CNC(C2CC3CCCCN3C2)=O)CC2(CC2)CN1C(C1CCCCS1)=O Cc1sc(Br)nc1C(N1CCCCC1C)C(=O)NCC1CCCO1 N1(C(c2ccc(C)o2)=O)CC2(CCN(C(=O)CN3CCc4ccsc4C3)CC2)C1 CC1(C)CCN(C(c2sc(Br)c(Cl)c2Cl)=O)CCS1=O N1(C(C=Cc2n(CC)ccn2)=O)CCN(C)C(CNC(=O)CN2CCCC2C)C1 C12(C(=O)NC3C(OC)C(O)C3)COC(C1)C(NC(c1cc(C(N)=O)co1)=O)C2 N1(C(c2cc(C)c(C)s2)=O)CC2CCN(C(c3cc(C(F)F)ccn3)=O)CC2C1 c1(CNC(C(C(C)C)F)=O)cnc2ccsc2c1 c1(NC(=O)CCCN(C)C)cc(Br)ccc1I.CC1CC2CN1C2 C1(CC(C)C)Oc2cc(Br)ccc2C1NC(N1CC(C)C(C)C1C)=O C(=O)(CC(O)CN(C)C)NC(C1C(C(=O)Nc2c(CC)csc2)C1)C CC(CCC(=O)NC(C)C(CO)NC(=O)CSCC(N)=O)N(C)C C(=O)(N=c1cccn[nH]1)C12C(C)(C)C1CN(c1ncnc3n[nH]cc13)C2 C1(NC(c2c(CC)occ2)=O)CCSC12CN(C(=O)C=Cc1ccc(=N)[nH]c1)C2 c1(C(=O)NC2C(NC(Cc3nc(C)c(C)o3)=O)CC2)cncc2c1CCC2 c1(CC(=O)NCC2CC(NC(C3(C4CC4)CC3)=O)C2)ccc(S(N)(=O)=O)cc1 C1(C(=O)NCCC(=C)CNC(C2(CC(F)F)CCC2)=O)CCn2cncc2C1 c1(C(N2C3C(C(=O)NCCCC4CC(C)C4)C(C3)C2)=O)ccnc(O)c1F C1(C2CC2)(NC(c2c(C)oc(C3CCNCC3)n2)=O)CCOC1 CC(=O)CCCC(=O)N1CC(NC(C2CC2C2CC2)=O)CC(C)C1 c1(CNC(C(CC)O)=O)nc2c(s1)CN(C(=O)CCCC(C)=O)CC2 c1(C(N2CCC(NC(C(C#C)(C)C)=O)C2)=O)ccc(N)c(F)c1Br C(=O)(C(C(C1CC1)OC)N1CCC(CCc2ccccc2)CC1)NCC(=C)C c1(C(c2nnnn2CC2CCOCC2)NCNS(N)(=O)=O)cn(CC2CC2)nn1 C(=O)(CNC(C1(CC(N)=O)CC1)=O)NC(C1(NCCO)CC1)C c1(C(N2C(CNC(=O)C=CBr)CCCC2)=O)ccc([N+](=O)[O-])cc1C(F)(F)F c1(-n2c(NC(C(=O)NCC(=O)NC3CCCC3)=O)ccn2)ccccc1Cl c1(C(=O)NCCC2CCC(NC(C(Cn3ccc(C)n3)C)=O)C2)cn(C)nc1O C12(C(=O)NCCc3c(C(N(C(CCC(C)C)C)C)=O)c[nH]n3)CCC(CC1)CC2 CN1C(=O)NCC1C(=O)NCC1(CNC(=O)COCC(F)(F)F)CC1 C1(NC(C2CC(NC(=O)CCc3ccccc3)C(O)C2)=O)CN2CCC1C2 C1(C)(CNC(C2C(CC)OCC2)=O)CCCN1C(=O)COc1cccc(O)c1 c1(C(N2CCC(O)(CNC(c3ccc(C#C)cc3)=O)C2)=O)ccc(C#C)c(F)c1 N1(C(CC2CCN(C(c3c(C(C)N)[nH]cc3)=O)CC2)=O)CC(C2CC2)C1C1CC1 C(C(CC(C)C)C(=O)NOCC(N1CC(CO)C1(C)C)=O)OC c1(OCC=C)c(C(=O)NCC=CCNC(=O)C=Cc2cn(C)cn2)cccc1C C(=O)(C(C)(C)CCCO)N1C(C)CN(C(c2cc(O)cc(O)c2)=O)CC1 N1(C(CC2(C)CC2)=O)CCN(C(=O)CN2CCCC2CO)CC1 N1(C(c2ccnc(Br)c2)=O)CC2(CCC(NCc3cnc(O)nc3O)C2)C1 N1(C(CC2N(C(c3c(C)n[nH]c3)=O)C3CCC2C3)=O)CC(O)C2(CCCC2)C1 C=CCC(C)C(=O)NC1CC(C(N2CC(C)(C#N)C2)=O)CC1O C#Cc1cccc(OCC(=O)NC2CN(C(=O)CCC(=C)C)C3CC23)c1 CC(CCc1ccccc1)CC(=O)NC1CN(C(=O)C(O)c2ccsc2)C1 CCCC(C(=O)N1CCCC1C1(NC(c2csc(CC)n2)=O)CC1)S(N)(=O)=O C(=O)(C(C)(C)C(F)F)NCc1nccc(C(=O)NC(C)Cc2cnccn2)c1 Cc1ncc(C(=O)NC2CC(CNC(C3CCCCCC3)=O)C23CCC3)c(C)n1 C1(NC(CC(C)F)=O)COC2(CCN(C(=O)CSC(F)F)CC2)C1 N1(C(C2(OC)CCCC2)=O)CC(C)OC2(CCN(c3cncc(C#N)n3)C2)C1 C1(CCC)CCCCC1(c1nnnn1C(C)(C)C)NCCCCO.c1(C2CC2)ccoc1 C1(NC(C2(COCC)CC2)=O)CC2C1CCN2C(c1cccc(C(F)F)n1)=O C=CCC(C(=O)N(C(C)C(=O)NCC1CCCN1C)C)C(C)C C1(C(N(C)CCc2ccccc2)=O)CCC2(CC2)N1C(C1CC(C)(C)C1)=O c1(C(=O)NCC(N(C)C(c2ncn(C)n2)=O)C2CC2)cc(Br)ccc1N c1(C(C(=O)NC(CCN(C(C=CCCC(C)C)=O)C)C)(F)F)cc(F)cc(F)c1 c1(C(N2CC(C(C(=O)N(CC(C)C(F)(F)F)C)OC)C2)=O)ccnc(C)c1N CN1CC(=O)NCC1C(=O)NNC(=O)c1ncon1 Cc1cc(C(N2CCCC(O)(CNC(C3CC(O)C3)=O)C2)=O)c2cnn(C)c2n1 c1(C(C)C)noc2ncc(C(N3CCC(C)C3CNC(=O)C3=CCCC3)=O)cc12 C(CCC(C)C(=O)NCCCC(C)(C)NC(C1CCCCC1(C)C)=O)OC Cc1nn(-c2ccc(F)cc2)cc1C(N1CC(CNC(=O)CO)C(C)C1)=O c1(C(=O)NC2C3CCN(C(C=Cc4cn(C)nc4)=O)C3C2)cnc2c(c1)CCC2 C(=O)(C(C)(F)F)N(C1CCN(C(C2CC(CF)C2)=O)C1)CCC CC1CC(N(C)C(c2cc(CNC(=O)Cc3cn[nH]c3)cs2)=O)CCO1 c1(C(=O)NC2CCN(C(C3C(C)CCO3)=O)C2)ccc(S(C)(=O)=O)o1 N1(C(CSC)=O)CCCC(O)(CCNC(=O)CCC2CC2C)C1 N1(C(C=C(C)C(F)F)=O)CC2OCCN(C(=O)C(C)N3CC(C)C3)C2C1 C(=O)(C(C(C)(C)C)NC(c1ccc(C2CC2)o1)=O)N(CCCC#C)C N1(C(C(C)CF)=O)CCC2(CCC2CNC(c2ncccc2N)=O)CC1 C12(NC(CC)=O)CCN(C(c3cccc(OCc4nc[nH]n4)c3)=O)CCC1C2 N1(C(c2cc(OC)ncc2)=O)C2CCC(C2)C1C(=O)Nc1ccc(I)cc1 c1(NC(N2CCN(C(C)C(F)(F)F)CC2)=O)ccc(Cl)nc1P(C)(C)=O C1(C(=O)NC(CC=C)CC=C)CCC(C)(C)N(C(=O)C=CC)C1 c1(OCC(=O)NC2(CC(=O)NC3CC3)CCC2)ccccc1CO CC1(C)CN(C(C2CC2(Cl)Cl)=O)CC1C(=O)NCC1(F)CC(O)C1 N1(Cc2cnc(C)s2)CCC(NC(=O)Cc2cccc(C(F)(F)F)c2)CC1C C1(C(C)NC(C2(C)CC(=C)C2)=O)CCCCN1C(=O)CCOCC(F)F N1(C(CC(C(C)C)NC(C23CC(F)(C2)C3)=O)=O)CC2(CCC(C)OC2)C1 C1(NC(C(CNC(=O)CC2CCCNC2=O)O)=O)CC2(CCOC2)C1 c1(C(N(C2CCCC2)CCNC(C2CCS(=O)(=O)C2)=O)=O)cc(Cl)c(Cl)s1 c1(OC)ccc(C)cc1NC(=O)C(CC1CC1)NC(=O)CC=C(Cl)Cl c1(C(=O)NCCCCNC(C2C(OCC)C2)=O)cc(Cl)c(F)cc1OC N1(c2nc(N(CC(=C)C)C)c3c(n2)ccs3)CCOc2ccc(F)cc2C1 CCC(CC(C)C)C(=O)N1CCOC(CN(C(=O)C(F)=C(C)C)C)C1 c1(C(=O)NC2(CO)CCN(C(C3CCCCS3)=O)CC2)cccc2nonc12 c1(C(=O)NC(CN(C(CCC(=O)OCC)=O)CC)CC)nn(CC)cc1[N+](=O)[O-] C#CCC(CC(F)F)C(=O)NC1CN(C(=O)CCCOC(C)C)C(C)(CC)C1 C1(NC(C(c2c(C)cccn2)(F)F)=O)C2CC(O)C1N(C(=O)CN(C)C(C)C)C2 C1(SCC(=O)NCC2CC(C(=O)N(C3(C(N(C)C)=O)CC3)C)C2)CCOCC1 c1(C(=O)NCC(C)(C2CCC2)NC(c2nnn(C)n2)=O)cc2ccc(F)cc2s1 C1(c2nnnn2-c2ccccc2Cl)(Nc2cccc(F)c2)CCC(=C(F)F)CC1 c1(C(=O)NCC(CNC(c2n(CC)ncc2)=O)C)c(C)cccc1[N+](=O)[O-] N1(C(CCOCC)=O)CC2ON=C(CNC(c3ncc(C(N)=O)cc3Cl)=O)C2C1 N1(C(c2snc(CC)n2)=O)CCC(C)C(C(F)(F)F)C1 c1(C(=O)NC(CC(C)NC(CNC(CC)=O)=O)C)c(C)cc(Cl)cc1C CC(C)CC(C)(C)C(=O)N(CC(O)CN(C)C(c1occc1C1CC1)=O)C Cc1ccc(CC(=O)NC2CN(C(=O)Cc3cc(F)ccc3Cl)CC2O)c(C)c1 c1(C(=O)NC(C)CNC(=O)CC2CSC2)c(O)nc(=O)n2c1CCC2 C1(C(=O)NCCCNc2c(CC)cccc2)CC2(CC2)CN1C(=O)C(C)N(C)C CC(C)CC(C)CC(=O)NC(C)(C)CN(C)C(c1cnc(C(C)(C)C)[nH]1)=O C(=O)(CC(CC)C(C)(C)C)NCC1N(c2nnc(CCC)s2)CCC1 N12CCOCC1SCCC2=O.C1(C(N(CCCOC)C)=O)CCCN1C(N)=O c1(OC)cc(C(=O)NCCCc2nc(C3CC3)cs2)cc(OC)c1C(=O)O C1(N(CC#C)C(C2CC2=C)=O)CCN(C(C2CCC(=O)C2)=O)CC1 c1(OC)cc(F)c(NC(C2CCCN(C(c3cccs3)=O)C2)=O)cn1 CC1(NCC2CCC(CNC(=O)OC(C)(C)C)CC2)CCC(=O)NC1=O C1(NC(c2cnc(C)o2)=O)CN(C(=O)C(c2c(C)n[nH]c2C)C)C2(CCCC2)C1 CC(C)(F)CCC(=O)NCC1CC1CNC(c1cccnc1S)=O c1(C(=O)NC(CC)CNC(=O)CCN2CCCC2)cc2cc([N+](=O)[O-])ccc2[nH]1 N1(C(Cc2n(C)ncc2)=O)CC2CC(C1)N(C(=O)CC1CC(C3CC3)C1)C2 c1(C(N(C(C)C(C)C)CCOC)=O)[nH]c(C)c(C(=O)COC(C)=O)c1C Cc1nn(C)c(C)c1NC(=O)NCc1ccc(-n2ncnc2C)cc1 C1(F)(CNC(=O)C(O)C2CC2)CCC(CNC(C2(O)CC2)=O)CC1 C1(C(=O)NCCN(C(=O)CN(C)C2CC2)CCC)CC(=O)OC1(C)C c1(C(N2CC3(C(NC(C(C)N(C)C)=O)CCS3)C2)=O)cc(F)cc2cnccc12 C1(CNC(C=C2CCC(C)CC2)=O)CC(C)CN(C(=O)CCN2CCC2)C1 C12(NC(COCC(=O)NC)=O)CCN(C(c3cc(COC)[nH]n3)=O)CC1C2 c1(C(c2nnnn2CC2CC2)NCC(CCC=C)(C)C)cn2cc(Br)ccc2n1 C1(C(=O)NCCN(OC)C)CCN(C(C2CC2C2CCC2)=O)CCO1 C1(NC(C2OCC(C)C2)=O)CC(=O)N(C2CN(C(=O)CCNS(C)(=O)=O)C2)C1 c1(C2(C(=O)NC(C)C(C)NC(c3coc(Br)c3)=O)CC2)ccc(F)c(F)c1 C(=O)(CCCCC(=O)NC1CCCCC1C(N1CCC(C(C)(C)C)CC1)=O)OC Cc1ccc(C(=O)NC2(CO)CN(C(=O)Cc3ccnn3C)C2)cc1 Cc1c(NC(c2cccnc2-c2cccc(NC(C)C)c2)=O)ccc(C#N)c1F N1(C(c2c(CC)c[nH]c2)=O)CCC(CNC(c2ccnc(S)c2)=O)(OC)CC1 NS(=O)(=O)C(C(=O)N1CCC(F)(CNC(=O)C=C2CCC2)C1)c1ccccc1 n1(CCC(=O)NCC2(NC(C3C(=C)C3)=O)CC(OC)C2)cc(Br)c(C)n1 CN1CC(C(=O)NCC(CNC(=O)CCc2cncs2)C(F)(F)F)CCC1=O c1(CC)nc(=N)[nH]cc1C(N1CC(NC(C2(C)CC(F)(F)C2)=O)C2CC12)=O c1(C(C)C)nn(C)cc1C(=O)N(C)CC1CCN(C(C2(C#N)CCC2)=O)CC1 S(=O)(=O)(c1ccsc1)NC(c1n(CC)cnn1)C C1(C(=O)NC2(C3CCCCO3)CC2)CCN(C(=O)c2ncccc2Cl)O1 C1(C(=O)NCCN2CCOCC2=O)CCC2(CC2)N1C(C1CC1c1ccco1)=O c1(C(=O)NCC(=O)OCC(=O)N(C2CCCC(F)(F)C2)C)c(F)cccc1Cl c1(-c2ncc(C(=O)NC3C(NC(CC(CC)C)=O)C3)s2)c(F)cccc1F C1(F)(C(=O)NC(CNC(C(C(C)C)N(CC)CC)=O)CC)C(C)(C)C1(C)C Cc1cccc2c(C(N3CCN(C(c4c[nH]c(C#N)c4)=O)C(C)C3)=O)coc12 c1(C(=O)NC2CCCN(C(C(CC)n3nccc3C)=O)C2)cc(C#N)ccc1F C1(CNC(Cc2ncc(CC)[nH]2)=O)CCN(C(C2(C)CCCC2C)=O)C1(C)C CN(C(=NCCF)NCC12CCC(C)(C1)OC2)CC1CNC(=O)O1 c1(SCC)ccc(C(N2CCC2CNC(C2ON=C(C)C2C)=O)=O)cn1 c1(CCC)[nH]nc(C(=O)NCC(C(C)(C)C)NC(C2CC2(C)C)=O)c1[N+](=O)[O-] c1(OC)cc2c(cc1C(N1CC3CCC1C(O)C3)C(=O)NC(C)C)OC(C)C2 CC1CCC(C)(C(N2CCC(NC(=O)C#CC(=O)N(C)C)C(F)C2)=O)C1(C)C N1(C(c2c(C)onc2)=O)CC(NC(=O)C(O)C2CCCC2)C2CCCC12 N1(C(C=CC(C)(C)NC(CC2(COC)CC2)=O)=O)CCCCC1CC(C)O C(CCN(C)C(C1(S(C)(=O)=O)CC1)=O)(C(C)C)NC(C1CCN(C(C)=O)C1)=O N1(C(C2C(C3(C)COC3)C2)=O)CCC(C2CC2)C1C(=O)NC(C(O)CO)C1CC1 N1(C(C(CC)C(C)C)=O)CCc2nc(CNC(=O)C(C)CC(C)O)sc2C1 C(C(C)(C)C(=O)NC1CN(C(C2CCS2(=O)=O)=O)C1)OC C=C(Cl)CCC(=O)N1CCOCC1CNC(=O)CCC1CC1(F)F N1(c2cc(C)ncn2)CCC(NC(c2csc(C3CCCO3)n2)=O)C(O)C1 CCC(CC(=O)NC1(C(=O)NCC2CC(F)(F)C2)CC(O)C1)C(C)C CC(C(=O)N1CCCC1)(C(F)(F)F)NC(c1cc2ccc(Br)cn2n1)=O C1(C)(CNC(C(CCSC)NC(C)=O)=O)CCN(C(=O)CNC(=O)C2CC2)CC1 c1(C(=O)NCCCOCCNC(CCCC(C)C)=O)ccc2c(c1)OCC2 Cc1cc(C2CC2)ccc1C(=O)NCC(C)NC(=O)C(C)Cc1c(C)noc1C C(=O)(N=c1[nH]nc(Cl)c2c1CCC2)ON.c12ccc(ccc1=O)cc2Cl C1(NC(c2cn(C(C)C)nn2)=O)C=CCN(C(=O)C(c2ncccc2F)(F)F)C1 C(N=c1nc2sccc2c(N2CCOCC(C)(F)C2)[nH]1)c1nn(C)nc1Br N1(C(C2CC(C)(O)C2)=O)CCN(C(c2ccc(O)nc2Cl)=O)C(CC2CC2)C1 N1(Cc2ncn(C)c2)CCCC1(C)C(=O)N(C1CC1)Cc1ccccc1 c1(CN2C(C(N3CC(C)(O)C3)=O)CC(F)C2)cnc2n1CCCCC2 CC1CCC(=CC(=O)NC2C=CCN(C(=O)Cc3cccs3)C2)CC1 C(=O)(C1CCc2nccn21)N1CC(OC)C(NC(c2nc(C)n(C)c2C)=O)C1 C(CC(C)C(=O)NCC1(C(=O)NC(Cn2cncn2)CC)CCCC1)=CCC N1(C(CN2CC(CCCCCC)C2)=O)CCN(C(=O)C2=CC(C)(C)C2)C(C)C1C C12(C(N3CC(NC(c4ccc(Cl)s4)=O)C3)=O)CCCC(CCC1)C2O C(=O)(C(C)CCCC(C)C)NCC(C)=CC(N1Cc2c[nH]nc2C1)=O Cc1ncc(Cl)c(C(=O)NC2CCCCC2NC(=O)C(C(C)C)n2cnnn2)n1 N1(C(CCCCCC)=O)CC2CCCN(C(=O)CCCc3ncc(C)o3)C2C1 c1(C(=O)NCC2(O)CN(C(C(C)c3ccco3)=O)C2)cncn(C)c1=O C=CC1CN(C(=O)C(C)(C2CC2)N(C)C(c2cn(CCOC)nn2)=O)C1 N1(C(C2C(C=C(C)C)C2(C)C)=O)CCOC2(C1)CN(C(c1c[nH]c(=N)c(C)c1)=O)C2 c1(C(N2C(C)C(C(=O)NCc3nn[nH]n3)CCC2)=O)cccc2[nH]ncc12 N1(C(C(C(C)O)C)=O)CCN(C(c2ccccc2C(F)F)=O)CC12CCC2 CC(C)C(=O)C(=O)N1CCN(C2CN(C(=O)CC3(O)CCC3)C2)CC1 N1(C(c2cn(C)nc2)=O)CCC2(CC1)CC2C(=O)NCC(c1ccccc1)F c1(NC(C(c2occ(C)c2)N(C)C(c2n[nH]c(C)n2)C)=O)cccc([N+](=O)[O-])c1 CC1(C)CC=C(C(=O)N2CC3CC(C2)CN(C(=O)CC(O)C2CCCC2)C3)CC1 c1(C(=O)NC2C(CNC(C3N(CC)CC3)=O)C2)ccc(C)c(Br)c1C C1(NC(C2C(NC(C3C(C)(C)OC(=O)C3)=O)CC=CC2)=O)Cc2ccccc2C1 c1(NC(C2N(Cc3c(OC)c(Cl)ccc3)CC2)=O)ccc2cn(C)nc2c1 C(=O)(C(C)(C)CCCNC(=O)CSc1nc[nH]n1)NCC1CCN(C(C)=O)C1 c1(C(=O)NCC2CCC2C(N(C2CCS(=O)(=O)C2)C)=O)ccc(N)cn1 NCCCC(O)C(=O)N1CCC(n2cc(-c3cn[nH]c3)nn2)CC1 c1(OC)cccc(CC(=O)NC(CNC(=O)C(C)SC)C(C)C)c1 N1(C(c2ccc(C(=O)OC)[nH]2)=O)CC(CNC(C2(Cl)CC2(C)C)=O)C(O)C1 C1(CC#C)(C(=O)NCC(F)CNC(c2cnn(C)c2OC)=O)CCOCC1 C1(C(=O)NC(CNC(c2nc(CC)sc2)=O)C(C)C)CCCOC1c1cn[nH]c1 c1(C(=O)OCC(C(CC)(C)C)=O)cc(Br)cc(S(C)(=O)=O)c1F C1(CNC(C2C(C=C)C2)=O)CCCN(C(c2ccn(C3CCCC3)n2)=O)C1 c1(OCC)cncc(C(=O)NC2CCN(C(=O)CC3(OC)CCCC3)C2)c1 c1(OC)cc(OC(C)C)ccc1N(C1CC2CCC(C1)N2)C(c1cc(C)[nH]n1)=O Cc1ccnc(CNC(=O)CC2CCN(Cc3ccc(C(F)F)cn3)C2)c1 C1(C(=O)NCCCC(=C)Cl)(CNC(C2CC(=O)C2)=O)CC12CCC2 C1(O)(CC(=O)NCC2C(CNC(COCC(=O)OC(C)(C)C)=O)C2)CCCOC1 c1(NC(CC(C)N(C)C(C2CC23CCOCC3)=O)=O)c(O)cccc1F Cc1nn(C(C)C)cc1C(=O)N(C1CN(C(=O)Cc2cncnc2)CC1O)C c1(C(=O)NC(C(C)NC(c2c(C)nc[nH]2)=O)C)cccc(Cn2cncn2)c1 CCCC(CCC)C(=O)NCC1CC(C)(C)CN1C(C1CCC1c1nc[nH]n1)=O c1(OC)cc(C)ccc1C(N1CCC(O)C(NC(C2(CN(C)C)CC2)=O)C1)=O c1(C(=O)NC2CN(C(c3cc(C)nn3C)=O)CC2O)ccc(C(F)(F)F)cc1C C1(C(N2C(CNC(C3CC3Br)=O)CC(OC)C2)=O)CCC2(CC1)CC2 C1(NCCNC(N(C)CCN2CCCCC2)=O)CCN(C2CCCCC2)CC1 c1(OC(C)C(=O)N(C)CCN(C)C(c2[nH]nnc2C2CC2)=O)ccccc1CO Cn1ccc(C(=O)NCC2CN(C(=O)C(=O)NCCC(N)=O)C2)cc1=O C(=O)(C(CCCC)C(C)C)NC1C(C(N(CCCC)C2CC2)=O)OCC1 CC(C)(C)CC(O)CC(=O)NCC1CCCN1C(=O)CSCC1CCCCO1 N1(C(C2C(CC)OCC2)=O)CCC(CCN(C(=O)Cc2cccnc2C)C)CC1 C1(C(=O)Nc2c(OC)cccc2)CN(C(=O)C(CO)OC)C(C)(C)C1 c1(C(=O)NC(CNC(C(C(C)(C)C)SC)=O)C(C)C(C)C)ccc2oncc2c1 c1(-c2cn(C3C(N4CCC(OC)C4)CCC3)nn2)cc2occc2s1 CC(C)CCCC(=O)N(C1CCCN(C(c2cocn2)=O)C1)CCF c1(C(=O)NC2CCCCCN(C(=O)Cc3ccno3)C2)cc(F)c(Cl)cc1Cl c1(OC)ccc(C(=O)NCC2CC(C(=O)N)OC2)s1.C1CO1.C1CO1.C1CO1 c1(OCC(=O)NC2C(NC(=O)CCCCCF)COC2)ccc(Cl)c([N+](=O)[O-])c1 C1(C(=O)N(C2CC2)Cc2ccccc2)COCCN(c2nnnn2-n2ccnn2)C1 C(=O)(C(F)C(C)(C)O)N1CC(C(N2CC(C(C)C)C2)=O)(CO)C1 C1(N(C)C)CCCN(CCC(=O)NCC(C)(C)CNC(=O)CC2(CO)CC2)C1 N1(C(=O)COCC2CCCC2)CCC(O)(Cn2cc(-c3ccccc3Cl)nn2)C1 N1(C(CSCC=C)=O)CCOC(CNC(c2ccoc2CCC)=O)C1 Cc1cncc(CC(=O)NCCNC(=O)C(C)Oc2ccccc2)c1 C1(C(N2CCC(CC3CC3)CC2)=O)CC2(CCN(C(C3CC(CF)C3)=O)C2)C1 c1(-n2cc(CCC#N)nn2)ccc(C(=O)NCC2CCOC2)cc1 N1(C(=O)Cc2ccccc2)CCN(C(C2CS(=O)C2)=O)CC1c1cn[nH]c1 C12(CNc3ncccc3C3CC3)CC1CN(OCC)C2 c1(C(=O)NC2CN(C(c3c(C)onc3)=O)CC2F)cnc2ccccc2c1 Cc1ocnc1C(c1nnnn1CC1CCCO1)NCc1csc(Br)c1 N1(c2cc(OCC)ncn2)CCC(NC(C2CCCN(C(N)=O)C2)=O)C(O)C1 C1(C(=O)NCC(CN(C)C(c2nnn(-c3ccccc3)n2)=O)O)COCC1(C)C CCCCC(C)C(=O)N1CC(OC2CCN(C(c3n[nH]cc3Cl)=O)CC2)C1 c1(CC)ccc2cc(C(N3CCC4(CCC4NC(=O)CC(F)F)CC3)=O)[nH]c2c1 c1(C(CNC(=O)C(Cl)=CCl)NC(C2CCC(C)O2)=O)ccc(C(C)C)cc1 Cn1c(C(N2CC(OCC(=O)NC(CCO)C3CCC3)C2)=O)cccc1=O N1(C(C=C(COCC)C)=O)CC2(CC(C(=O)NCC3CCC(CC)O3)CO2)C1 C1(CC=C)CCCN(C(C2(NC(=O)C(C)C3CCC3)CC(F)C2)=O)C1 Cc1ccc(OCCC(=O)NC(C)C(CO)NC(c2cccs2)=O)c(C)c1 C1(C(=O)NCC2(CC)CC2)(CO)CCN(C(c2cn(CC)cn2)=O)C1 CCCC(C(=O)NCCCC1CN(C(=O)CC(C)(C)O)CCO1)C(C)C CCC(C=O)NC(=O)C(O)CC.C(C)(C)(C)OC(=O)NCCN(C1CC1)C(C)C c1(-c2n(CC=C)c(N3CCC(C)(C(N)=O)C3)nn2)ccc(Br)cc1F C(CCC(C)CC(=O)N1CCC(NC(c2n[nH]c(C)c2Cl)=O)CC1)=C(C)C CCC(C(=O)N1CCCC(C(N2CC3(C)COCC3(C)C2)=O)C1C)C(C)(C)CC N1(C(c2cc(C)n(C)c2C)=O)CC2(CCC2)CC1C(=O)NCCC(O)C(F)F c1(CNC(CC(CC)C)=O)ccc2c(c1)NC(=O)C2=O.C12COCCN(C1)C2=O C1(C(CC(C)C)NC(C(=O)N(CC)CC)=O)CCCN(CCc2ccccc2)C1 c1(N(C(C(C)(C)C)=O)CCO)ccc(Nc2c(CN3CCCC3)cccc2)cc1 c1(C(=O)NCCCCNC(=O)Cc2csc(C3CC3)n2)cc(O)c2sccc2c1 CC1(C)CC(CC(N2CCOC3CC23)=O)N(C(=O)C(CO)NC(N)=O)C1 C1(c2n(CC=C)nnn2)(NC(C)Cc2cccs2)CC2(CCC(C)(C)CC2)C1 Cc1cc(C#N)cnc1C(N1CCC2CC12C(N1CC(O)(c2cnn[nH]2)C1)=O)=O c1(C(=O)NCC2(F)CCCN(C(C3C(C#N)C3)=O)C2)ncn2c1CCCC2 N1(C(CC(C(C)C)O)=O)CC(CNC(=O)Cc2nncn2C)OC(C)(C)C1 c1(C(N2CCC(NC(C3(c4cc[nH]n4)CCC3)=O)C2)=O)csc(C(F)F)n1 c1(OC)cc(C)c(S(=O)(=O)NC2(C(F)F)CCOC2)c(C)c1 c1(C(=O)NCC(CC)NC(c2nn[nH]c2C(F)(F)F)=O)c[nH]c(=NC)s1 n1(CC)c(NC(C2CC(=O)NC(=O)C2)=O)nc2cc(Cl)ccc12 C1(N(C)C(C2C=CCCC2)=O)CCC2(CC1)CCN(C(c1cc(Cl)n[nH]1)=O)C2 c1(C(=O)NC2C(NC(C(CCOC)C)=O)COC2)cc(Cl)c(Cl)cc1N Cc1cccc(F)c1CC(=O)NCCCCCCN(C)C(C1CCCN(C)C1)=O C1(NC(C=Cc2cnc(C)s2)=O)CC2CC(NC(c3cc(C(C)C)[nH]n3)=O)C1C2 CC1(C)CCC(CNC(C2CC2CNC(C2CSC2)=O)=O)OC1 C1(NC(COc2ccc(C)cc2Br)=O)CN(C(=O)CNC=O)CCC12CCC2 n1(CC(=O)NCC2CCCN(C(C(CC)C#N)=O)C2)cc2ccccc2n1 c1(C(=O)Nc2ccc(SCC)cc2)c(F)ccnc1Cl c1(C(C)C)cc(C(=O)NCCOCCCN(C(=O)Cc2cncn2C)C)n(C)n1 CC1(C)C(C(=O)NCC(C2CCC2)NC(c2ccnc(OC3CC3)c2)=O)C1(C)C C1(N(CCC)C(c2n[nH]c(COCC)n2)=O)CCN(C(=O)C(C)CC)CC1 C#Cc1cncc(C(=O)N(C2(CC(N3CCN(C)C(CC)C3)=O)CCC2)C2CC2)c1 c1(C(=O)NCC(C)N(C(=O)C(F)C2CC2)C)cc(F)cc2ccoc12 N1(C(CC(CC)C2CCC2)=O)CC(C)C(C)(C(=O)NCC2CC23CCOCC3)C1 C=CC(F)(F)C(=O)N1CC(O)(CCNC(c2ncccc2C2CC2)=O)C1 C=CCC(CC(C)C)C(=O)NCCC1(C(=O)NCC2(CSC)CCCCC2)CC1 CC(C)(C)C(CNC(c1ccsc1C#N)=O)C(=O)NCC1C=CCOC1 C#CCC1C(=O)N1.C(CO)(C(C)CC)NC(=O)CSCCC C1(F)(C(=O)NCC2N(C(=O)CCn3ccnn3)CCC2)CC2(CCC2)C1 C(N=C(NC1CCC1)N1CCN(c2ncccn2)CC1)C1C(CC)C1 C#CCC(C(=O)NC1CC(C)(NC(C2(c3ccccc3Cl)CC2)=O)C1)C1CC1 c1(C(=O)NCC2OCC(CNC(C(N)=O)=O)C2)coc2cc(O)ccc12 C1(CC(=O)NCc2nnn(CC)n2)CCN(C(=O)CC(C)C)CC1 N1(C(CNC(CC)=O)=O)CCC(C(F)(F)F)C(NC(c2oncc2C)=O)C1 c1(C(c2cccs2)C)cn(C2CC3(C(=O)N(CC(C)(C)C)CCO)CC23)nn1 C=CCC(CC(C)C)C(=O)N1CCC(N(C(=O)CCC2CCCC2)CC)C1 c1(NC(C)=O)cnc(C)c(C(N2CC(CNC(c3ccn(C)n3)=O)C2)=O)c1 C1(NC(C2CCC(CC)CC2)=O)CN(C(c2cc(N)cc(N)c2)=O)CC1(C)C C1(C(N(C)CC2CN(C(CC(C)c3ccccc3)=O)C2)=O)CC(=O)N(C2CC2)C1 C1(NC(C2CCC2)=O)CCC(O)CN(C(=O)CC2C=CCC2)C1 C(=O)(C(C)(C)CCCNC(c1c[nH]c(=N)o1)=O)Nc1cn(CC)nc1 CC(C)C(F)(CNC(C1CC(F)(CF)C1)=O)C(=O)NC12CCN(CC1)C2 c1(C(c2cc(O)nc(S)n2)NCc2n(CCC)ccn2)ccc(C)c(Br)c1O CCCC(CCCNC(=O)CCCc1nncn1C)NC(C1(CO)CC1)=O N1(C(c2nn(C)c(Br)c2)=O)CC(C2CN(C(=O)Cc3cccs3)C2)C1 C(=O)(CCCC(N)=O)N1CC(C(C)NC(c2cn(CC(N)=O)nn2)=O)C1 C(=O)(CC1CCc2ccccc21)N1CC=CC(NC(C2(C)CC2(F)Cl)=O)C1 CCCC(CC)C(=O)NC(CNC(c1c(F)cccc1Cl)=O)C1CC1 c1(C(=O)NC23CCN(C(C(C)S)=O)CC2C3)ccc2c(=N)[nH][nH]c2c1 c1(C(N2CCC(CNC(c3c(C(C)(C)C)ocn3)=O)C2)=O)cnn2ccncc12 C(=O)(C(C)CS(C)(=O)=O)NCC(CCCC)NC(=O)C(CC)CC C1(CCN(C(=O)CSc2ccncc2)C)CCCCN1C(C1CCCNC1=O)=O N1(C(C2CCC(NC(Cc3ccn(C)n3)=O)C2)=O)CCN(CC(F)(F)F)CC1 c1(N(C)CC=CC2CC2)ccc(S(=O)(=O)N2CCCC(CF)C2)c(Br)c1 N1(C(c2ccn(C)n2)=O)CC=CC(NC(C2CC(=O)N(Cc3ccco3)C2)=O)C1 C1(C(=O)OCCSCc2ccncc2)CCC(=O)N(CC(F)(F)F)C1 Cc1ccc(C(=O)NC(CCF)C(=O)NC23CCN(CC2)CC3)nc1C O=C(C#CC1CCC1)NCC=CCNC(=O)CCc1ccc(Cl)nc1 C1(C(N2CC(NC(=O)COCc3ccnc(O)c3)C(O)C2)=O)(CC)CCCCC1 N1(C(c2cnc(C)o2)=O)CCC2(CC(C(=O)Nc3cccc(CCF)c3)C2)C1 Cc1cc(C(C)C(=O)NC2CCCCC2NC(=O)Cc2cn[nH]c2)cc(C)c1 N1(C(c2ncc(CC)s2)=O)CCCCC(NC(c2cccc(O)c2F)=O)C1 C1(C(=O)NC2(CCC)CCC2)CN(C)CCN1C(C1OCCCC1(C)C)=O c1(SCC(N2CCC(C(c3cn(C4CC4)nn3)C)C2)=O)cccc(C#N)c1 c1(NCC2C(NS(C)(=O)=O)COC2)[nH]c(=NC2CCCCC2F)nc2sccc12 C1(C(=O)NCCCC(=O)NCCSCC)CCOC(C)C1 C1(CN(C(=O)CN2CCCCC2)C)CCCN(C(C2CCC(=O)NC2)=O)C1 C1(C(C)C)(C(=O)NC(C)C(C)F)CCCN1C(C1CC1C1CC1)=O c1(C(c2cn(CC(C)NC(c3ccc(CC)s3)=O)nn2)O)ccc(F)cc1 C1(NC(CC(=C=C)C)=O)CN(C(=O)CN2CCOCC2)C(C)(CC)C1 N1(C(C2(C=C)CCOCC2)=O)CC(CNC(=O)CC(C)(C)C#N)C2(CCC2)C1 c1(C(=O)NC2C(NC(c3cc(C)nc(O)c3)=O)C2)cnc(O)c2ccsc12 N1(C(C(C#C)(C)C)=O)CCC(C)C(N(C)C(C2OCCCC2(C)C)=O)C1 N1(C(C(=O)NC2C3(CN(C(C)=O)C3)CCC2)=O)CCC2(CC1)CNC(=O)O2 C1(CCCC)CCC(C(=O)NCCCNC(=O)C(C2CCC2)OC)CC1 C1(NC(Cc2n(C)ccn2)=O)CCCC(NC(C2CC(=C3CCC3)C2)=O)CC1 c1(C(=O)NC(C(C)C)CNC(=O)CNC(=O)CCCCO)nc(Cl)ccc1F N1(C(CN(CCC)C)=O)CC2(CCC(NC(c3c(Cl)cc(Cl)cc3Cl)=O)CC2)C1 C1(NC(=O)CN2CCCCCC2)CC1C1CCN(C(=O)C(F)OC(F)(F)F)CC1 c1(CNc2c(C(=O)NCc3cc(C)ncc3)nccc2)c(O)ccc(Cl)c1Cl C=C(C)CCC(C)NC(c1cc(CNC(=O)C(C)n2cccc2)[nH]n1)=O c1(CNC(c2cn(CCCCC)nc2C)C)ccc(Cl)c2cccnc12 C1(CNC(c2c(C(C)C)scn2)=O)CC(C)N(C(=O)C(O)C2CC2)C1 Cc1cc(-c2cnn(C)n2)ccc1Br N1(C(CC23CC(C)(OC2)C3)=O)CC2(CCCN(C(C3CC4(C3)CC4(F)F)=O)C2)C1 C1(CNC(=O)CC2CCOCC2)CC2(CCCC2)CO1.C12CCN(CC1F)C2=O C1(C(=O)NCCOCC(C)(C)O)CCCCC1(C)NC(C1CCOC1C1CC1)=O N1(C2CN(C(=O)NCC3=CCCC3)C2)CCCS1(=O)=O C1(NC(=O)OC)CCC2(CCCN2C(=O)NCc2ccc(C(=O)OCC)o2)CC1 C1(CN(C)C(c2ccoc2Br)=O)CCCC(NC(c2cncnc2)=O)C1 CC1(F)CCCCN(C(C2CC(O)CCN2Cc2ncc(Cl)nc2Cl)=O)C1 Cc1noc(C)c1C=CC(N1CCC(C(C)NC(=O)Cc2cncn2C)CC1)=O c1(C(C)C)ccc(C(=O)NCC2CC2CNC(=O)CC2(N(C)C)CCCC2)o1 C=CCC(CC(=O)NCC(C)CC(=O)NC)NC(C1(CO)CC1)=O C1(CC(=O)NC2(CNC(C3CC4CC4C3)=O)CCCC2)CCCCO1 c1(CNC(C2CCOCC2)COC)nc(C)cn1C N1(C(c2c(C)c(F)cnc2)=O)CCC2CN(C(=O)CCc3cncs3)C2C1 c1(OCC)cnc(C(N2CCC(N(C(=O)C(C3CCCCC3)F)C)CC2)=O)cn1 C#CCC(O)C(=O)N1CCN(C(=O)Cc2nonc2C)CC1 N1(C(c2cnn(CC)n2)C(=O)NCC)CCC(C#N)CC1 c1(NCC2(COC)CCC2)[nH]c(=NCC2(S(C)(=O)=O)CCCC2)nc2scnc12 c1(OC)nccc(C(=O)NC2CC(NCc3c(F)cccc3F)C2)c1F C1(C(=O)NC2CC(CNC(c3cccc(NC)n3)=O)C2)CNC(=O)CC12CCC2 C(CC(CC)C(=O)N(CC(C)C(=O)N1CCC(C(CC)CC)C1)C)=CC N1(C(CC)CC)CC(C(N2CC(CCNC(=O)COCCCOC)C2)=O)CC1=O CC(C)CCCC(=O)N1CC(C)(OCC(N2CC(CO)CCC2C)=O)C1 CCCCCCC(C)C(=O)NC(C)(CSC)C(N1CCC2CC1C(=O)O2)=O c1(C(N2CCCN(C(C(c3ccn(C)n3)(C)C)=O)CC2)=O)ccn2c1CCCC2 n1(CCCOC)c(N2CCCC(c3nc(C)no3)C2)nnc1C1CCCCN1C N1(C(c2cccc(C)c2F)=O)C2CCC1CC(NC(C1CC3CC1CC3O)=O)C2 C1(C(N2C(CC=C)CCCC2)=O)CCN(C(=O)CC2OCCO2)CC1C C(C(C)(C)CNC(=O)C(C1CCN(C(c2cnn(C(C)C)c2)=O)C1)C)OC C(C)(CSC)(C(=O)Nn1cnnc1C)NC(CC(CCC)O)=O C1(C(C)C)CCC(C(=O)N(C)Cc2nnn(C)n2)N1C(=O)OC(C)(C)C Cc1cnnc(C(N2CC(O)(CNC(=O)CCOCCN(C)C)C2)=O)c1 Cn1nc(CC(N2CC(NC(=O)C(C)(O)C3CCOC3)C2)=O)cc1C(F)(F)F N1(C(CC(C)(F)F)=O)CCC2(C)CN(C(=O)CC3CC3(Cl)Cl)CC12 N1(CCCCCNC(COCCCCCC)=O)CCCC(C(N)=O)C1 n1(CC)c(C)nn(CC(=O)N(CC(C)NC(C2(C)COC2)=O)C)c1=O C(CCN=C(NCC1(OC)CCCS(=O)(=O)C1)N1CCC(S(=O)(=O)NC)C1)OC c1(SC)cccnc1C(N1CCC(C(C)NC(=O)CN2CCOCC2)C1)=O N1(C(C2CN(C)C(=O)N2)=O)CC2CCCC(NC(=O)CCC3CC3(Cl)Cl)C2C1 C1(NC(=O)C2=COCCC2)CC2(CCN(C(c3ccc(C(O)CF)cc3)=O)C2)C1 N#Cc1ccc(CNC(C23CC2CN(C(=O)C=Cc2ccc(O)cc2)C3)=O)nc1 Cc1cc(-n2cc(-c3cnn(C)c3CNC(c3ccc(F)s3)=O)nn2)cc(F)c1 c1(C(=O)NCCC2CCN(C(CCCCNC(N)=O)=O)CC2)ccc(F)cc1Cl N1(C(CCCCC=C)=O)CCCCC2(CCN(C(=O)C(C)COC(C)=O)C2)C1 S(=O)(=O)(c1ccc(C(=O)NCC(C)OC)c(Cl)c1)NC1(C)CN(C(=O)NCC)C1 c1(C(=O)NC2CCCN(c3nc(C#N)cc(C)n3)C2)cccc2ccncc12 c1(-c2nc(C(C(C)(C)C)N(S(=O)(=O)C3CC3)CCC)on2)cccnc1F CC(N=c1[nH]c(N(S(C)(=O)=O)CC2CCC2)nc2cccc(F)c12)c1ccoc1 c1(OC)ccc(C(N2CC3C(NC(c4ccn(C)n4)=O)C3C2)=O)nc1 C1(NC(c2cc(CCC)ncc2)=O)C2CCN(C(=O)Cn3ccnc3C)CC12 C1(NC(CCN(C(C(C)C)=O)CCCO)=O)CCCC1(C)N(C)C Cc1cc(C(N2CCN(C(c3n[nH]c4c3COC4)=O)C3CC23)=O)n2ncnc2n1 C1(N(C(=O)CCSC2CCC2)C(C)C)CCCCCC1 Cc1[nH]nc(C(=O)NC2(C)CCN(C(=O)CCC3CCCN3C)C2)c1Cl Cn1ncc(C(=O)NCCCCC2CN(C(c3cnc(C(C)(C)C)s3)=O)C2)n1 N1(c2ccnc(NC3C(C(C)C)OCC3)n2)CCOCC(OC2CCCC2)C1 CC1CN(C(C2(F)CCCOC2)=O)CC1NC(c1nccn1C)=O N1(C(=O)Cn2cnnn2)CCC(NC(C2CC(n3cnnc3)C2)=O)C(CO)CC1 C1(C(N2C(C(=O)OC)C=CCC2)=O)CN(C(c2nn(C)cc2C)=O)CC1(F)F C(C(F)(F)C(=O)NCC(C)(C1CC1)NC(C1CC(C)CCO1)=O)OC Nc1cccc(CC(N2CCCC2CCCNC(C2CC3CC2C3)=O)=O)c1 C1(C(=O)N(C)C)CCN(c2nc(C(C)C)cc(C)n2)CCC1NC(C(CC)SC)=O C(c1ccc(O)cc1)=CC(N1CCC(OCCNC(C2CCC(C)C2)=O)CC1)=O C(C(CC(=O)N(C1CC2CC2C1)C)NC(C1CC=CCO1)=O)OC c1(C(=O)NC(CNC(C(C)C(F)F)=O)C(C)(C)C)cccn2cncc12 C1(CNC(C(CC)C)=O)(OC)CCN(C(C2(OC)CCSC2)=O)CC1 N1(C(CC2N(C)CCCC2)=O)CCc2c(c(CNC(=O)CC3CSC3)nn2C)C1 C(=O)(CC(C)(C)C(=O)N(CCCCN(C)C(C1(C)CC1(F)Cl)=O)C)OC C1(C(C)(C)C)C(NC(=O)CNc2nccs2)CCN1C(=O)CC1CCC(=O)NC1 C(=O)(CCCCCNC(C)=O)NCCC1CN(C(C=CCOC)=O)CC1C N1(C(CCC=C)=O)CC(C2(Nc3nc(C(F)(F)F)ns3)CC2)C1 c1(C(=O)NCC2CC(NC(=O)COCC3CCCO3)C2)cnc(Br)o1 Cc1ncccc1C=CC(N1CCC1CNC(=O)CC(O)C1CCCC1)=O C(=O)(CC(C)(O)CCC)NCc1c(CNC(CN(CCC#C)C)=O)cccn1 CN=S(C)(=O)c1ccc(C(=O)N(C(C)CN(C(=O)CCn2ccnc2)C)C)cc1 Cc1ccc([N+](=O)[O-])cc1C(N1CC(NC(=O)C=CC(C)(C)C)CC1C)=O N1(C(c2ccc(C(F)F)o2)C(=O)NC(CC)C)CCOCC(O)C1 c1(-c2cn(C(COC)COC)nn2)cc2c(s1)CCN(C(=O)Cc1cnn(C)c1)C2 c1(CNC(=NCC)NCc2cnc(C3CC3)o2)ccc(C)c(C#N)c1 C1(n2cc(-c3cc(C)nnc3)nn2)CC2(C1)CC(C(C)C(N1CCCSCC1C)=O)C2 CC1=C(C(=O)NCC(F)CNC(C2CCCCN2C)=O)C(C)(C)CCC1 c1(C(=O)NC2CCC(CNC(c3csnc3Cl)=O)C2)ccc(=O)n(C2CC2)c1 C12(C(=O)NC(CC(C)C)CNC(c3ccc(C4CC4)o3)=O)CC3CC(CC1C3)C2 c1(C(=O)NCC(CCC)NC(=O)CC(CC)C(C)C)cnc2cc[nH]c2c1 C1(CNC(CCCC=C)c2nnnn2CC2CCOCC2)CCC(C)(C)CC1 C1(CC(N2CCC(O)(C(C)C(=O)NC(=O)C(C)(C)C)C2)=O)CCC(C)(O)CC1 c1(C(C)(C)NC(=O)OCc2cnc(C3CCC3)s2)ccc(C(F)(F)F)cc1 N1(C(c2c(CC)c[nH]n2)=O)CCCC(NC(c2cccnc2F)=O)C1C c1(C(=O)NC2CC(n3cc(C(CC)(O)CC)nn3)C2)cnc2c(c1)COCC2 c1(C(=O)NC2C(CNC(c3c(C#C)c[nH]n3)=O)COC2)ccc2ccoc2c1 N1(C(C2(C(=O)OC)CC2)=O)CCCCC(CNC(C2(C)CC3CCC2O3)=O)C1 c1(OC)ccc([N+](=O)[O-])c(NCC2CN(C(C3CC34CCSCC4)=O)CCO2)n1 C1(CNC(C2CC3(CCC3)CO2)=O)CCC2CN(C(=O)Cc3ccsc3Cl)CC12 C(=O)(C(C)CC(C)(C)C)NC1C(F)CCN(C(COCCCC(C)C)=O)C1 c1(C(=O)NC2(CO)CCCN(C(COCC(C)C)=O)C2)ccc2c(c1)CNC2=O Cc1nc[nH]c1CNC1CC(C(=O)Nc2ccnn2CCN(C)C)C1 Cc1scc(C(=O)NC(C(=O)NCC(c2nncn2C)C)C2CCCC2)c1C Cc1cc(Cl)ccc1C(=O)NCC1CCCC1NC(=O)CC1COC(C)(C)C1 CC1(C)CC(CNC2CC3C=CC2C3)CCO1 c1(C(=O)OC)cnc(C(=O)NCC(C2CC2)N(C(=O)C(O)C2CCCC2)C)cn1 C1(C(=O)NC2CC(NC(=O)CC3(n4cccn4)CC3)C2)COc2ccccc2O1 C(=O)(CS(F)(F)(F)(F)F)N(C1CCCN(C(=O)C2=NOC(C)(C)C2)C1)C c1(C2C(C(N3CCC(CCNC(=O)CCc4ncco4)C3)=O)C2)ccccc1Cl Cc1cn2cc(C(=O)NC3(CCNC(=O)CC4CCC(C)(O)CC4)CC3)sc2n1 C12(CNC(C(=O)N(CC(C)(C)C)Cc3ccc(Br)cc3)=O)COCCN1CCOC2 c1(C(=O)NCCCN(C(=O)C(C)NC(C(C)(C)C)=O)CC)n[nH]cc1C(F)(F)F C(=O)(C#CC1(C)CCCO1)NCC1(CC)CCC1.c12ccc(cc1)o2.C1C(=O)N1 c1(CC)cc(C(=O)NC2CC(C)(CNC(=O)C(CC)SC)C2)oc1CC N1(C(COC(CC)(C)C)=O)CC2CC(O)C1C2NC(=O)CCn1cc(C)cn1 CCN=C(NCc1ccc(Br)cc1)NCc1cn(C(C)(C)C)nn1 c1(OC)cc(NC(=O)CCOC2CN(C(=O)C=CCN3CCC3)C2)cc(Cl)c1 C1(NC(c2ccc(C)c(Cl)c2)=O)COC2C(NC(=O)C(C)OCC(C)C)COC12 c1(OCC)c(OC)cc(C(=O)NCCC(O)CNC(=O)C=CS(C)=O)cc1OC c1(CC)nc(C)oc1C(=O)N(C)CCOCCCNC(C1CCCSC1C)=O CC(=O)CCCC(=O)NC1CCCN(C(C2CCCNC2=O)=O)C1C C1(C(=O)NCCC23CC(C)(OC2)C3)CCc2ncc(Br)n2C1 C(=O)(C(C)(C)CCSC)N1C(CC)C(NC(c2csnc2C)=O)CC1 Cc1nnc2cnc(C(N3CC(CNC(C4C=CCC4)=O)OC(C)(C)C3)=O)cn12 c1(C(=O)NCC2(O)CCN(C(Cn3ncc(CC)c3)=O)C2)ccc(OC)c(Cl)n1 C1(C(N(CCN(C(=O)CC2CCCNC(=O)C2)CC)CC)=O)CCCC1C1CC1 C1(CCC)(NC(=O)C(COC)NC(=O)CN)CCN(C(C2CC2(Cl)Cl)=O)CC1 N1(C(C2CN(Cc3ccccc3)CC2(F)F)C)CC(C)Oc2ccncc21 C[Si](C)(C)C1(CNC(C2CCC(NC(c3ccc(F)s3)=O)CC2)=O)CC1 C(=O)(CC(C)CC(C)(C)C)N1CC2CCN(C(c3cc(C)[nH]c3C)=O)C2C1 c1(C(=O)NCC2(F)CC(NC(c3cc(C)oc3)=O)C2)nc(C(C)C)oc1C CCC(CC(F)(F)F)C(=O)N1CCCC(C2CCCCN2C(C2SCCS2)=O)C1 N1(C(CNC(=O)OCC)=O)CCC(C(=O)NC2CCN(C)C2(C)C)C(O)C1 N1(C(CC2(CSC)CC2)=O)CCC2CCCC12C(N1CCC(n2cnnn2)C1)=O c1(N2C(C3CCN(C(C(COC)(C)O)=O)CC3)C(C)(C)C2)ncnc2ccsc12 c1(OC)cc(C(N2CCN(C(=O)Cc3cscn3)C3CC23)=O)c2ccccc2n1 C1(N(C(CC(C)SC)=O)C(=O)C=C(C)C(C)C)CCCN(CC(C)C)C1 N1(C(Cc2cc(C)no2)=O)CCN(C(=O)C(C)S(N)(=O)=O)CC1C1CC1 Cc1cnc(C(=O)NC(c2cn(-c3cc(F)ccc3F)nn2)C)cc1C c1(OC)ccc(Br)c(CNC2CC(C)CN(C(C34CCC(CC3)CC4)=O)C2)c1 S(=O)(=O)(c1ccc(N(C)CCN(C)C)c(Br)c1)NCC1(C)CCC(C)CC1 C1(N(C(C(C)SCC)=O)CCOC)CCN(C(=O)CC2CC=CCN2C)CC1 Cc1nc(O)ccc1C(=O)NC1CN(C(c2c(C)noc2C(F)F)=O)CCC1C c1(C(N2C(C(C)NC(=O)CCc3nc[nH]n3)CCC2)=O)ccc2ncsc2c1 C1(CC=C)(NC(c2cnn(CCO)c2)=O)CCN(C(=O)C(C(C)C)N(C)C)CC1 Cc1cc(NCCCCO)ncc1S(=O)(=O)N1CC(c2ccccc2)OCC1C CCCCC(C)(F)C(=O)NCC1CN(C(c2cn3nc(C)sc3n2)=O)CC1(C)C C#Cc1cnc(C(N2CCOC(CCCNC(c3c[nH]nc3Cl)=O)C2)=O)c(C)c1 Cc1ccc(CCC(=O)N(c2nccs2)C(=O)COCc2ccncc2)nn1 Cc1nnc(CC(=O)NC(C)(CNC(=O)CC(O)C2CCCC2)C2CC2)o1 Cc1cc2scc(CC(=O)NCC(C3CCC3)NC(=O)C=Cc3cncs3)c2s1 CC1CCc2nc(C(=O)NCCN(C(c3cnn[nH]3)=O)C3CC3)ccc2C1 c1(N(CC(CC)O)C)ccc(S(=O)(=O)NCc2c(C)nn(C)c2C)c(Br)c1 c1(C(C(=O)NC(C)CNC(C2CC2(F)F)=O)O)ccc(Cl)cc1F CC(N=c1[nH]c(=NCCc2c[nH]nc2Br)[nH]c2c1CSC2)C1CCC(F)(F)CC1 C1(CNC(CN2CC(C)C2)=O)N(C(c2ccc3scnc3c2)=O)CCCC1(C)C Cc1cc(C(N2CCC(N(C(=O)C(C)SC(C)C)CCO)C2)=O)c(C)s1 CCC(C)(O)C(O)C(=O)NCCc1cccc(C)c1C N1(C(c2c(CSCC)cccc2)=O)CC(C)C(NC(=O)Cc2cccs2)C(C)C1 c1(OC)ccccc1C1(C)CC1C(N1CC2CC1C2NC(=O)CCOC(C)C)=O c1(CC(=O)NCC2N(C(c3c(C)ccnc3)=O)CC(F)C2)ccc2nonc2c1 c1(OC(C)C)ccc(NC(C2CC3(C2)CN(Cc2ccccc2I)C3)=O)cc1Br c1(C(=O)NC(C2CN(C(=O)C3=NNC(=O)CC3)CCO2)C)ccc(Cl)c(F)c1O Cc1ncc(C(=O)Nc2cccc(NC(=O)CC3CCCC(=O)N3)c2)cc1N c1(OC)cncc(C(N2CC(C(C(=O)NC3CCC(C)(C)C3)OC)C2)=O)c1 C(C(O)CNC(=O)C(C)N(C(=O)C(OC)OC(C)=O)CC)OCC C1(CCC)(NC(C(C)=CC)=O)CCN(C(=O)C(=Cc2ccccn2)C)CC1 Cc1cc(F)c2c(c1)CCN(C(=O)CCc1cccc(F)c1Cl)C2 C1(C(=O)NC(CC)CCO)CC2(CCN1C(c1cncc(OC)c1)=O)CC2 CCC(C)(C(=O)N(CCCNC(c1csc(-c2cccc(Cl)c2)n1)=O)CC)OC c1(C(N2CC(C(N)=O)(CNC(C3C(C)COCC3)=O)C2)=O)c(F)ccc(F)c1Cl N1(C(C(c2cncnc2)C)=O)CC2(CCC2)CC1C(=O)NC1COC(C(F)F)C1 CC(CC(F)F)C(=O)NCCN(CCOCCO)C(c1c[nH]nc1C1CCCO1)=O CCC(C)(CNC(C1(F)CCCN(C(c2cc(OC)ns2)=O)C1)=O)C(N)=O c1(OC)cnccc1C1(C(=O)NCC(C)CO)CC(N)C1 C(=O)(C(F)(CNC(C1(C(C)C)COC1)=O)C(C)C)NCC1(C#C)CCCC1 c1(NCC=C)nc(N2CC3C(C2)C3(C)C)nc2c1ncn2CC C12(NC(c3n(CC)ccn3)=O)CCN(C(=O)Cn3ncnn3)CCC1C2 C1(CC)CN(C(c2cnc(Cl)s2)=O)CCC1NC(c1cn(CCOC)nn1)=O C(=O)(CCC(C)(C)F)NC1C(NC(C=Cc2ncn(C)c2)=O)C1 C1(NC(CC=C)=O)CN(C(c2ccc(Cl)c(OC(F)(F)F)c2)=O)CCC1(F)F c1(C(N(C(CC)CC(=O)NC2COC(C(F)F)C2)C)=O)cccc(C)c1N c12ccc(F)cc1CNC2=O.C1(C(=O)OC)CCCC1C(=O)Nc1nccs1 C(=O)(C(O)CSC)NCC(CC)NC(=O)C=CCOC C(=O)(CCC1CCc2ccccc21)NCC(CNC(C#CC1(C)CC1)=O)(C)O c1(C(=O)NCC2CN(C(C(C(C)C)O)=O)CC2C)cccc2c1CCCC2 CC(C)(C)CCC(=O)C(=O)N1CCC(CF)(NC(c2cc3ncccn3n2)=O)C1 c1(CC(=C)C(=O)NC(C)CCC=C(C)C)ccc(F)cc1F N1(C(c2cc(C)ncc2C)=O)CC2(C1)SCCC2NC(=O)C(O)C1=CCCCC1 c1(-c2n(CCCO)nc(-c3cncc(Br)c3)n2)ccc(Cl)cc1Cl N=c1sccn1CC(N1CC(O)(CNC(C2CC(=O)N2)=O)C1)=O Cc1ccc(C(=O)NC(C)(CNC(=O)CC2CCSC2)CO)cc1O CCC(C)(C)C(=O)NC12CC1CN(C(C1(c3cncnc3)CCCC1)=O)C2 c1(C(CNc2nnc(-c3ccc(Br)o3)s2)OC)cccc(C)c1 c1(C(N(C2CCCC(NC(C=CCCC)=O)C2)C)=O)cc(C)c2[nH]nnc2c1 C1(NC(CN(C)C)=O)CCCC1NC(=O)C(CO)NC(=O)Cc1ccccc1 c1(C(N(CCCNC(=O)C(O)COC)CC)=O)cn2cnnc2cn1 c1(OC)cc(C(=O)NC2CC(CNC(=O)C(C)O)C(O)C2)c(F)cc1Br c1(C(N2CCC(NC(CCCn3c(C)nc(C)n3)=O)C2)=O)ccn2c1CCCC2 CCCCCCC(C)C(=O)N1CC2(CCN2C(c2cc(F)n(C)n2)=O)C1 C1(N(C(c2c(C)nco2)=O)C)CCCCC1N(C)C(c1n[nH]cc1Cl)=O Nc1nccnc1C(N1CCCCC1C1(NC(=O)CN2CCCS2(=O)=O)CC1)=O Cc1nc2ccc(F)cc2c(NC2(C)CCc3ccccc3C2)c1C C(=O)(C(C)(F)C(C)(C)F)NCC(CC(C)C)NC(C1CCCC2CCCN12)=O N1(C(CCC(C)OCC)=O)CCC(NC(=O)CCC(C)N(C)C)C2(CCC2)C1 CS(=O)(=O)c1ccc(C(N2C3CCC2CN(C(=O)CCN2CCC(F)C2)C3)=O)o1 C1(CNC(CCOCC)=O)COCCN(C(C2CCCCNC2=O)=O)C1 C(=O)(CC(CN(C)C)C(F)F)NCCCN(C(=O)CN(C)S(N)(=O)=O)CC N1(C(C(CCC)OC)=O)CCC(C2CC2NC(c2nsnc2O)=O)CC1 C1(C(N(CC(=C)C)C)=O)C=CCN(C(C2CCCC2CCC)=O)C1 C1(C(N2CC(CCC#C)C2)=O)CC2CCC1N2C(=O)CC1CCC(C(C)C)CC1 N1(C(CC(C)n2ccnc2)=O)CC2(COC(CNC(=O)Cc3ccsc3)C2)C1 N1(C(CCOCC)=O)CC(C(=O)NC(C)CCC(=O)OC)CCC1(C)C N1(C(C(n2cc(-c3ccc(CCC)cc3)nn2)C)=O)CCC2CCC(C1)S2 C#Cc1ccccc1C(N1CC(NC(c2cc3sccc3s2)=O)C(C#N)C1)=O c1(CC(N2CCC(N(C(C(CN(C)C)O)=O)C)C2)=O)cccc(Cl)c1F c1(NCC=CCNC(c2c(CCC)occ2)=O)cc(C)nc(COC(C)C)n1 N1(C(C2CC(C)(CC)C2)=O)CCCCC(NC(c2csc(-c3cnc[nH]3)n2)=O)C1 C(=O)(CCCCCCN=[N+]=[N-])NC1CCN(C(c2cc(C)ncc2)=O)C1C c1(OCC(=O)NCC(C2CC2)NC(C2CCCOC2)=O)cncc(Br)c1 C1(C(=O)NCC2(NC(c3cc(Cl)no3)=O)CC2)CCCN(C(c2cncs2)=O)C1 c1(C(=O)NCC(C(C)C)NC(C2C(OC)(OC)CC2)=O)ccc(NC=O)cc1 c1(COCC)ccc(NC(=O)NCC2CN(C)CCN2C)cc1C C(=O)(CCCCC(=O)NC)N1CC(CNC(C(CCCC)O)=O)C1 c1(C(=O)NC2CCC(CN(C)C)CC2)ccc(N)c(-c2nccs2)c1 C1(NC(C(COC)NC(c2cnc(Cl)nc2C)=O)=O)CC2(CCC2)CO1 CCCCCC(CC)C(=O)NCCC1CCCN1C(c1ccc(CC)nc1C)=O Cc1ncc(C(N2CC(C(N3CCC3CN=[N+]=[N-])=O)CC2(C)C)=O)c(=N)[nH]1 C12CC3CCC1N(C3)C2=O.C1(C2CC2)(CNC(CNC(CC)=O)=O)CCC1 c1(C(=O)NCC2CCC(NC(C(CC)(CC)OC)=O)C2)cnc2ccc(C)cn12 C1(NC(C(c2cccs2)NC(C(CN(C)C)O)=O)=O)CC2CC1C(O)C2O C#CCC(C(=O)NCCC1(CNC(=O)CSCC(C)C)CC1)C1CC1 c1(SC)nc(C(F)F)cc(=NC2CCOC(C3CCCCN3CC3(Br)CC3)C2)[nH]1 C1(C(=O)NC2CC(NC(CSCCC(C)C)=O)CC2O)CCC([N+](=O)[O-])CC1 N1(C(C2N(C(c3c(C)nccn3)=O)CC(O)C2)=O)C2CCC1CC(C)C2 C=CC(C)(CCOC)C(=O)N1CCCN(C(=O)C(C)OCC(C)C)CC1 N1(C(CNC(C)=O)=O)CCC2(NC(C3C4CCC3(C)C4(C)C)=O)CCCCCC12 C1(=O)C(C)(C)CCc2cn(nn2)CCSC2CN1C2.c1(CC)nccn1CSC C(=O)(C1CCc2nccn21)N1CC(C#C)N(C(c2cncc(NC)c2)=O)CC1 C1(C(C)(C)NC(=O)C(F)C2CCC2)CN(C(=O)CC=C(Cl)Cl)CCO1 c1(C(C)SCCN2CCOC2=O)c(F)cccc1F Cc1ncc(CC(N2CC(CNC(C3CCC(=O)N3)=O)C(O)C2)=O)c(O)n1 c1(C(=O)NC(CNC(Cc2onc(CC)n2)=O)C(C)C)cc([N+](=O)[O-])ccc1O c1(OCC(=O)NC2CC3CN(C(CCCCC)=O)C2C3)ccc([N+](=O)[O-])c(C)c1 CC1CN(C(c2ccc(C#N)cc2)=O)CCC1NC(=O)C(C1CC1)C1CC1 c1(SC)nc(N2CC(C)(C)CC2CNC(c2ccncc2Cl)=O)cc(C(F)F)n1 C1(NC(c2cc(OCC)no2)=O)CC2CCC(C1C)N2C(C1CC2CCCC12)=O c1(C(=O)NCCC(=O)NCCCCCC=C)c(C)ncnc1C C(=O)(C1(C)CCc2ccccc21)NC1CC(NC(c2cn(C)nn2)=O)C(O)C1 N1(C(CC2CC(=C)C2)=O)CC(NC(c2ccc(OC(C)C)cc2)=O)C(C2CC2)C1 C1(NC(C(N2CCC(O)CC2)C)=O)CCOCC1NC(c1nc(C(N)=O)cs1)=O N1(C(CCC#C)=O)C(C(=O)NC2(c3ncc(C)o3)CC2)CCC1C N1(C(c2c(C)ccnn2)=O)CCN(C(c2ccns2)=O)C2CCCCC12 c1(C(=O)NCCCCn2cc(C(CC)O)nn2)ccc(OC)c(F)c1C(F)(F)F CCC(C(=O)N1CCC(CO)(NC(=O)Cc2cccnc2)C1)C(C)(C)CC C=CC1(CC(N2CCCC(NC(=O)CN3CCCCCC3)C2C)=O)CCCCC1 N1(C(=O)NCc2nccc(N)c2)CCCCCC1c1ccccn1 CN1C(=O)NCC1C(=O)NCC1CC1CNC(c1ccccn1)=O C1(CCCC)CN(C(=O)CC2CC(=O)NC2=O)CCN1C(c1cn(CC)cn1)=O C1(CNC(C=COCC)=O)CC(C)(C)CN1C(c1cnn(C)c1N)=O Cc1c(Br)cc(Cl)c(NC(C2CCN(C(c3ccc[n+]([O-])c3)=O)CC2O)=O)c1Cl C1(NC(c2nn(C)c(F)c2)=O)CC2CCC1CN2C(=O)C=Cc1ccco1 C1(NC(c2cn(C)nn2)=O)CCCCN(C(C2(N(C)C)CCCCC2)=O)CC1 c1(C(N2CC(OC)C(NC(c3cc(C(C)C)no3)=O)C2)=O)cc(C)ccc1F C1(CNC(C(C)OC)=O)CC(F)(F)CN1c1nc(C(=O)OC)ns1 C1(C2CCN(C(=O)Cc3ccncc3Cl)C2)(NC(c2cc(C)c(C)nc2)=O)CC1 C1(CC(=O)OCC)CCN(C(c2cc(C(C)(C)O)on2)=O)C1(C)C c1(C(CC)C(=O)Cc2csc(N3CCOCC3)n2)cc(F)cc(Br)c1.N1CCC1 c1(C(=O)NCC2N(C(C(C=C=C)C)=O)CCCC2)cc(O)nc2[nH]c(=N)ccc12 C(=O)(C(F)(F)C(C)O)NC1C2CC(NC(C3(CSC)CCC3)=O)CC21 c1(C(=O)NC2CC(NC(CCCSC)=O)CC2O)cc(C)c(F)cc1Cl c1(C(=O)NC2C(CNC(c3c(C)cc(CO)o3)=O)CCC2)cccc(F)c1N c1(OCC)ccc(C(CO)NC(c2cnn(C3CC3(F)F)c2)=O)cc1 c1(C(=O)NCC(CNC(c2c(C)n(C)nn2)=O)(C)C)n[nH]c2c1CCOC2 C(=O)(C1CCCn2nccc21)NCC1CCN(C(C(C=C)(C)O)=O)CC1CC O=C(C#CC1CCC1)NCC1CCCC1NC(c1cnn(-c2ccncc2)c1)=O C1(NC(=O)CCc2ccsc2Br)CCCCC1NC(C1C2CCCC12)=O N1(C(CN2CCN(C(c3csc(C)c3C)=O)CC2)=O)CCC(O)C(F)C1 C1(NC(=O)Nc2ccc(-c3cn(C)nc3)cn2)CCC2CCCC2C1 c1(C(N2CCN(C)C(CNC(=O)C=CS(C)=O)C2)=O)ccc2cnccc2c1 C1(NC(Cc2onc(C)n2)=O)CN(C(c2cn(C3CCOC3)cn2)=O)CCC1C C1(CNC(CC(=O)NC)=O)COCCN(C(=O)C#CC2CC2)C1 c1(C(N2CC3N(C(C(C)Oc4ccccn4)=O)C3C2)=O)cc2cc[nH]c2cc1Cl c1(NC(C)=O)cccc(NC(=NCC2CC2(Cl)Cl)NCC2CCCO2)c1 c1(C(N(C)CC2CCN(C(c3ccoc3Br)=O)C2)=O)cc(N)cc(O)c1 C1(NC(=O)CSc2ccncc2)CC12CCN(C(c1ccc(Br)c(F)c1)=O)CC2 C(C)(CCC(=O)NCC(CC1CCCC1)C(=O)N(C1CCCCC1O)C)OCC CC(C)(C)C1=NOC(C(N2CC(CNC(C3CC4C=CC3C4)=O)C2)=O)C1 N1(C(COCC(=O)OC)=O)CC2C3CCC(C2C1)N(C(=O)C(C)OCC(C)C)C3 C1(CNC(C(C)=C2CC2)=O)CC2CCC(C1)N2C(=O)CNC(=O)CCC1CCCC1 Cc1ccc(C(N2CCN(C3CCC(NC(C4CC(F)C4)=O)CC3)CC2)=O)cc1 c1(C(N2CCC(NC(C3C(CC)C3)=O)C2C2CC2)=O)ccc(=O)n(C)n1 c1(N2C(=O)C2)ccccc1C.c1(SC)nnc(-c2ccc(O)cc2)n1CC(N)=O C(=O)(CS(=O)(=O)CC(F)(F)F)NCC1CCN(C(CC(=C)C)=O)CCC1(F)F Cc1oc(CCN)nc1C(N1CC(n2cc(Cc3ccccc3)nn2)C(C)C1)=O c1(C(C(=O)NC(CC)CN(C(=O)CCc2cn[nH]c2)C)O)ccc(C)cc1 C(=O)(C(Cc1ccco1)NC(=O)C(C)n1cccc1)N(CC(COC)C)C c1(CC(=O)NCCC2CC(NC(c3c(C)cc(CC)o3)=O)C2)c(F)cccc1F c1(C(C(=O)NCCC(=C)CNC(c2cnc(SC)s2)=O)C)ccc(OC)cc1 CC(C)C(O)C(=O)N1CCC(OCCNC(C2(c3cccs3)CC2C)=O)CC1 C(CCCC(=O)N=c1ccn(C2CC2)[nH]1)NC(C1N(C)C(=O)CCC1)=O C1(NC(C(C2CCOCC2)OC)=O)CCCC1CNC(C1(F)CCC1)=O C1(C(=O)Nc2cc(OC)c(OC3CCCC3)cc2)CCCN2CCCCC12 c1(CCC(=O)NCC2CC2NC(c2nc(Cl)sc2Cl)=O)c(F)cccc1Cl C1(CC(=O)NCC(C)(CNC(c2ccc([N+](=O)[O-])[nH]2)=O)OC)CCC2(CC2)CO1 C(=O)(C(C)(F)C(F)(F)F)NCCOC1CCN(C(c2cc(CC)oc2C)=O)C1 c1(C(C)=O)cc(C(=O)NC(C(=O)NCC2(CC(C)C)CC2)C2CC2)n[nH]1 C(=O)(CS(=O)(=O)CCCC)NC1CN(C(C(F)=CCC)=O)C(C)CC1 C1(CNC(CC=CCNC(CC2N(C)CC=CC2)=O)=O)CCC=CCCC1 N1(C(c2c(N)ccc(Cl)n2)=O)CCc2nc(CNC(=O)CCC3CCC3)sc2C1 C=CCC(C)(O)C(=O)NCc1ccc(CNC(c2ccc(C(C)C)o2)=O)c(F)c1 c1(N2CC(CCOC)(NC(C3CCN(CC#C)CC3)=O)C2)nc(C)nc(O)c1C C12(NC(c3cc(C(N)=O)oc3)=O)CCCCC1CN(C(=O)C(N)=O)C2 C1(NC(C2(COC)CC2)=O)CCC(CNC(=O)Cc2scnc2Cl)C1 CC1CCCn2c(C(=O)NC(C)CCNC(=O)CNC(c3ccncc3)=O)cnc21 CCC(CC)C(C(=O)NCCN(C(C1CCCC1)=O)Cc1ccccc1)OC C1(CC=C)(NC(C2CC(Cl)(Cl)C2)=O)CCN(C(=O)Cc2ncncc2Cl)CC1 c1(C(N(CC(CN(C(=O)CSCCC#N)C)O)C)=O)ccnc(S(N)(=O)=O)c1 C12(C(=O)NCCC(=O)NCC(COC)O)C=CC(CC1)C2 C1(C(=O)NC2(C[SH]=C)CN(C(=O)C(C)C(C)CCC=CC)C2)CC2(CCCCC2)C1 C(C)(C(CC(=O)NC1CC(C(C)C)C1)NC(C1CCOC1(C)C)=O)OC C(=O)(CC(CC(C)C)NCC1CCC(c2nc[nH]n2)O1)OCC CC(C)C(C)C(CNC(=O)CCCCCF)NC(=O)Cn1ccc(C2CC2)n1 C(CC(=O)Nc1c(C)nn(CC)c1C)(C(F)F)NC(c1cccc(CC=C)c1)=O c1(OCC)ccc(NC(C2CN(C(=O)C(=O)NCC3(C#N)CCCC3)C2)=O)cc1 CC1CCC(CC(=O)NC2CCCC2NC(=O)Cc2cc(Br)cs2)C1 S(=O)(=O)(c1ccc(F)cc1)ONC(C1C(C)CCN1C(=O)C1=CCCSC1)=O C12(NC(C34CC(C)C3C4)=O)CCCC(CN(C(c3cocn3)=O)C1)C2 C1(CN)CCN(C(c2cn(Cc3ccc(-n4ccnc4)cn3)nn2)=O)C2(CC2)C1 C1(NC(c2c(C)scc2)=O)CCCN(C(C2(C)CCC(=O)C2)=O)CC1 c1(OCC)cc(N2CCN(C)CC2CNC(=O)C(C)N(C)C)ccc1[N+](=O)[O-] C1(C(=O)NCCc2c(C)ncs2)CCC(C(C)C)N1C(C1CS(=O)C1)=O C12(NC(Cc3ccc(CC)cc3)=O)CCCC1N(C(C1(C)C=CCCC1)=O)CC2 c1(C(=O)NCC2N(c3ncc(OCC)cn3)CC(F)C2)ccc(C)c(Cl)c1F C1(NC(c2cn(CC=C)nn2)=O)CCCCC12CCCN(C(C1(C)CC1)=O)C2 C1(CC(=O)NC2CC(CNC(CCCNC(C)=O)=O)C2)CCC(C)(C)O1 C1(NC(CCc2ccn(C)c2)=O)CCCC(NC(=O)CN2CCCNC2=O)C1 C12(COC)COC(C(N3CC(O)(C(C)NC(=O)C(C)c4cccs4)C3)=O)(C1)C2 N1(C(c2ccc(OCC)cc2C)=O)CC(C)CN(C(=O)COCC2CC2)C(C)C1 c1(CC=C)cccc(CC(C(=O)OCC)NC(=O)NC(C)C2CC2)c1 Cc1nscc1CC(=O)N(CCCN(C)C)CCNC(=O)C=CBr C(=O)(CCCCC1CC1)NC1CC(C)(NC(C(C)OC)=O)C1 C1(OCC(=O)N(CCCCNC(=O)Cc2n[nH]cc2Br)C)CCC(F)(F)CC1 c1(CCC)noc2nc(C)cc(C(=O)NCC3(NC(=O)OC(C)(C)C)CCC3)c12 c1(SCC)ccc(Br)c(C(c2nnnn2CC)NCc2ccc(C)cc2F)c1 c1(C(=O)NC2C3CN(C(CC(C)OC)=O)CC32)ccc(F)c(Cl)c1 C1(C)(CNC(C2N(C(C3C(CCC)CCC3)=O)C(C)C2)=O)CSC(C)=N1 C(=O)(C(CCOCCO)NC(C1CC(N(C)C)C1)=O)NC(C1CC(F)(F)C1)C#C c1(C(=O)NCC2(NC(C3CC(CCC)C3)=O)CC2)ccc(CC)cc1O N1(C(C2CC(OC)C2)=O)CCC(CCNC(c2ccc(Br)o2)=O)C1 c1(N(C)CC2CCN(C(=O)C=Cc3ccccn3)CC2)nc(Cl)nc2[nH]ccc12 c1(OCC)ccc2cc(CN3CCN(C(C)C)C(C)C3)ccc2c1 Cc1cc(C(=O)NC2(CC=CC(=O)NCCCS(C)=O)CCC2)cc(C#N)c1 C1(NC(c2n[nH]c(CC)c2Br)=O)CCCN(C(=O)CC=C(C)C)CC1F CC1C(=O)N1C.C(CCO)(C1CC1)NC(=O)C1CC1.c1(C=O)ccco1 C1(NC(C(CC)OCC)=O)COCCN(C(c2coc(C(F)(F)F)n2)=O)C1 CCN=c1cc(C(=O)NCC2CC(NC(=O)C(n3nc(C)cc3C)C)C2)cc[nH]1 N1(C(CSCCC(C)C)=O)CCC(NC(C2CCC(C)(C)CO2)=O)C(CO)CC1 c1(C(=O)NC23CC(CNC(C4CCCOC4)=O)(C2)C3)occ2c1CCCC2 C(=O)(C(O)CC(C)C)N(C1CCN(C(c2cc(C)ncn2)=O)C1)CCO c1(C(N2CC(CNC(C(n3c(C)cc(C)n3)C)=O)C(C)C2)=O)cc2n(n1)CCO2 C=CCC(C)(C)CC(=O)NCC1CCCN1C(=O)CCc1cccc(C(F)F)c1 c1(C(=O)NCCC2CN(C(c3ccsc3Cl)=O)CCO2)c[nH]c2nc(F)ccc12 N1(C(c2cncc(C)c2)=O)CCC(CNC(=O)C(C)OCCC(C)C)C(F)(F)C1 c1(C(=O)NCC2(OCC)CN(C(C(C(=C)C)(C)C)=O)C2)cccc([N+](=O)[O-])c1 N1(C(C=CCCC)=O)CCN(C(c2cc(Cl)c([N+](=O)[O-])[nH]2)=O)C(C)C1C c1(C(=O)NC2CC3CC(NC(C4C(C)C4C)=O)C3C2)cc(Cl)cc([N+](=O)[O-])c1O Cc1cccc(C)c1OCC(=O)N(C)CCNC(=O)CNS(=O)(=O)c1cccs1 N1(C(c2cccc(Cl)c2)=O)CCC2(C1)CN(C(C1CC=CCC1)=O)CCO2 C(CN=c1[nH]c(N(C)Cc2ccccc2)nc(=N)[nH]1)(c1ccccc1Cl)N(C)C C1(CNC(CC2(OC)CN(C(c3nc(O)sc3C)=O)C2)=O)CCCC12CCC2 c1(-c2nc(CCCN(C)C=O)nn2C2CCCC2)ccc(C#N)cc1N.C(C)(C)C n1(CC)nc(C(N2CCc3nc(O)nc(O)c3C2)=O)c2ccccc2c1=O C(=O)(C(C)C(C)NC(=O)C(CCC1CCC1)NC(=O)CC1CCCCN1C)OC N1(C(CC(C(C)C)O)=O)CC(NC(=O)COCC2CCCC2)C2(CCC2)C1 N1(C(C(C)C)=O)CCC12CN(Cc1cnc(Cl)cn1)C2 O=C(CCCCCCCC1CC1)NC1CC2(C1)CC2NC(c1ccc(O)cn1)=O N1(C(C2C(C)CC2C)=O)CCCC2(C1)CN(C(=O)C1=NOCC1)C2 N1(C(C(=O)NCC(F)F)=O)C(CC(=O)O)CCC1C1CC1.C(=O)(C(=O)N)N(CCO)C c1(OC)cc(N2CC(OCCNC(C3CCC(C)(CC)O3)=O)C2)ccc1[N+](=O)[O-] c1(C(=O)NC2CC(CNC(Cc3cc(CC)no3)=O)C2)cc2scc(Cl)c2[nH]1 CCCCC(C)C(=O)N1CCCC1(C(=O)NCc1cccc(CO)c1)CC CC1CN(c2ncc(Cl)cc2[N+](=O)[O-])CCC12CCOC2 CC1(C)CC2(CC(NC(=O)NC3CCCCC34CCC4)C2)C1 c1(C(=O)NC23C(C)OC(CNC(=O)C(C)(C)F)(C2)C3)cc(Cl)c(N)c(Cl)c1 c1(SCC)ccc(C(N2CCCCC2CNC(=O)CN(C)CCO)=O)cn1 C(C(C)C(F)(F)F)N(C(C(Cc1ccco1)NC(C1N(CC)CC1)=O)=O)C c1(OC)cccc(CN(C(=O)NCc2ccc(F)cc2O)C)c1Br C1(C(=O)NC2CN(C(C3(O)CCCC3)=O)CC2F)CC2(C1)CC(O)C2 c1(C(N2CC(CNC(=O)CC(F)(F)F)OCCC2)=O)ccc2c(c1)CCCC2 C(=O)(CCCN=[N+]=[N-])NCC1CCN(C(C(OC)OC)=O)C1 c1(CC)ccc(OCCC(=O)N(C(C)CNC(=O)C=Cc2sccc2C)C)cc1 c1(CCC(=O)NC2C(NC(C3N(C)C(=O)CC3)=O)C2)ccc([N+](=O)[O-])cc1Cl c1(CN(C(c2cnn(C)c2C(C)C)C(=O)NC)C)ccc(OC)c(Br)c1 c1(C(N(CCC(C)NC(C(C)OC2CCCC2)=O)C)=O)c[nH]c2nc(Cl)ccc12 Cc1ccc(C)c(C(N2CC(O)(CNC(c3ccnc(C(F)F)c3)=O)C2)=O)n1 N1(C(C2CC(SC)C2)=O)CCOC(CNC(c2c(CO)n[nH]c2C)=O)C1 c1(CC)nn(C)cc1C(=O)NC1CC12CC(NC(c1ccc(CO)cc1)=O)C2 C12(C(=O)NCC(CC#C)(C)CO)CCC(CN(C(=O)C(C)NC(=O)NC)C1)C2 c1(-c2cn(C3CCCN(C(N4CCC5CC5C4)=O)CC3)nn2)ncc(Cl)cc1Cl c1(C(=O)NCC(CC)NC(=O)CC2CSCCS2)coc2c1COC2 c1(C(=O)NC2CC(NC(c3c(O)ccc(CC)c3)=O)C2)cccc2ncc(C)n12 C(=O)(CCCCCS(N)(=O)=O)N(CC(CN(C(C(CCCC=C)(C)C)=O)C)O)C Cc1cc(F)c(C(C)C)cc1Nc1cn(C(C)(C)C)nn1 N1(C(CC2(C)CC(F)(F)C2)=O)CC(NC(c2ccn(C3CC3)n2)=O)CC2(CC2)C1 N1(C(Cc2ccc(OC)cc2)=O)CC(C)(C)C(NC(=O)C2=CCC2)C(C)(C)C1 c1(CCCN(CCCO)C(C)C)cnc(-c2ccccc2)[nH]1 c1(C(N(CC(C)NC(CS(CC)=O)=O)C)=O)c(OC)cc(OC)c(Cl)c1N c1(OC)ccc(C(N2CCCC(CN(C(=O)C(F)C(C)C)C)C2)=O)c(C)c1 CC(C(CO)NC(=O)Cn1nccn1)NC(=O)C(F)(F)C1CCOCC1 N1(C(CN(C(C(CCCC)F)=O)CCC)=O)CC2CCC(O)C(O)C12 N1(C(c2cc(OCC)n[nH]2)=O)CCCCCC(NC(c2cccc(N)c2C)=O)C1 C1(CNC(C2CCS(=O)(=O)C2)=O)CC(F)CN1C(c1ccc(C(F)F)cc1)=O Cn1cc(C=CC(N2CCC(N(C(C3CCCOC3)=O)CC3CC3)CC2)=O)nn1 C1(C)(CNC(c2c(C)oc(Cl)n2)=O)CCCN(C(C23CC4CC2C3C4CO)=O)C1 C1(NC(c2ncn(C(C)C)n2)=O)CC(C(=O)NCC2(CN=[N+]=[N-])CC2)C1(C)C Cc1cncc(CCn2cc(CN3CCOCC3C3CCOC3)nn2)n1 N1(C(C(C2CCN(C(=O)C#CC3CC3)CC2)C)=O)CC(CO)OCC1C c1(C(=O)OCC)n[nH]c(=NCC2c3ccccc3CN2C)o1 C=C(C)CCCC(=O)NC1CCCCCC1C(=O)N(C1CCN(CC)C1)C n1(CC)nc(C(=O)NC(CCOCCO)C(=O)N2CC(COC)C2(C)C)cc1O c1(CN(CC)CC2CCN(C(c3cnc(C4CC4)o3)=O)C2)nc(CC)cs1 c1(CC(=O)OC(C23CC(CCC)(C2)C3)=O)ccc2scnc2c1 c1(OC)c(C)cc(C(=O)NC2(C)CCN(C(C3(COC)CCCO3)=O)C2)cc1C C1(N(C(=O)N)C(n2cccc2)C)(CC23CC(CC(F)F)(C2)C3)CCOC1.CC(C)O C(C(F)(F)C(F)F)OCC(C)C.C1CC(=O)N1CC1CN(C(=O)CNC2CC2)C1 C1(NC(=O)CC2CCC=CCC2)CCN(C(=O)CCOCC(F)(F)F)CC1OC c1(OCC)ccccc1C(=O)NC(C(=O)NC1CCCCC1)C1CCOC1 C1(C2CC2)(NC(c2c(SC)n(C)nc2)=O)CCN(C(=O)C=Cc2nccs2)C1 N1(C(COCC)=O)CCOCC12CCN(C(=O)C1CC1)C2 C1(C(=O)NCCS(CC)=O)CN(C(=O)CSC)CC12CCC2 c1(C2N(C(N=c3cnn(COC)[nH]3)=O)CCC2)c[nH]c2ccccc12 CC#CCCCC(=O)NC1C2CC1N(C(=O)Cc1ccc(F)c(F)c1)C2 C1(C(N2CC(C)(C)C2)=O)CC12CCN(c1ncc(Br)c(C(F)(F)F)n1)C2 C1(CNC(C2C(C)C2)=O)CN(C(=O)Cc2ccc(F)nc2)CCC12CCC2 N1(c2n(CCOC)c(-c3ncnn3C(C)(C)C)nn2)CCC2(CCO2)C1 C(=O)(C(CCCCc1ccccc1)N(C1CCCC(C)C1)C)NCCSC C1(CCC)C(=O)N2CC1C2=O.c1(C(C)OC(c2n[nH]cc2Br)=O)cccc(F)c1 c1(OC(C)C)ccc(COc2ccc(-n3ccnc3)nc2)nn1 N(C1CCc2ccc(Br)cc21)C(C1CN(Cc2cc(I)ccc2F)CCC1O)=O N1(C(c2cc(OCC)no2)=O)CCC(C)C(CC(=O)NC2(Cl)CC2(F)F)C1 c1(C(=O)NC(C(C)C)CCN(C)C(C2CC2C(C)O)=O)cnc2sccc2c1 c12cc3cc([nH]c3cc1OC)CN1CCC1C(=O)O2.c1(COCC)ccccc1 O=C(C1Cc2ccc(F)cc21)NCCCOCCNC(c1ncoc1C1CC1)=O c1(OCCC)ccc(C(=O)NC2CC(CNC(c3ccccc3)=O)C2(C)C)cc1 N1(C(CC(=C)Br)=O)CCC2CCN(C(c3ccc(S(N)(=O)=O)o3)=O)CC12 Nc1c(F)ccc(F)c1C(N1CC2CCN(C(C3CCCCNC3=O)=O)C2C1)=O c1(C(=O)NC2C(NC(c3cc(CC)ncc3)=O)COC2)c(C)ncn(C)c1=O Cc1nc2cccc(C(=O)NC3CCCCC3NC(=O)C(C)OCC3CC3)c2s1 c1(CCNC(C2C(CNC(c3scc(C)c3)=O)OCC2)=O)cccc(O)c1 N1(C(CCCCCC)=O)CCC2(CCC(NC(c3cc(C)no3)=O)CC2)C1 c1(C(c2nnnn2Cc2cccs2)NCC(=C)Br)c(C2CC2)cnn1C N1(C(c2cc(C)ccn2)C(=O)NC(CC)(C)C)CC2(CCC2)C1c1ccccc1 C(=O)(C(O)P(C)(C)=O)NCCCC(C)NC(CCn1ncc(C)c1)=O C(CC(C)CC)(C(=O)N(C)Cc1ccnn1C)NC(C(C)=CCC)=O C1(C(N2CC(C)N(C(C3CN(C4CCOCC4)C3)=O)CC2)=O)CCC2(CCOCC2)C1 c1(C(N2CC(C)C(C)(CNC(=O)Cn3nnc(=N)[nH]3)C2)=O)ccc2cnnn2c1 C1(C(N2CC(=C)C2)=O)C(COC)CCN1C(=O)C1=CCSC1 Cn1nccc1CCCNC(=O)C(Cc1cc[nH]n1)NC(=O)CCC1CCOC1 Nc1c(C(N2CC(CNC(c3c(Cl)cccc3Cl)=O)C2)=O)cc(Cl)cc1F C1(CCNC(Cc2n(C)cnc2)=O)CCN(C(c2ccsc2)=O)CCC1(F)F N1(C(c2c(C)cccn2)=O)CC2CC1CN(C(=O)CC=CC(C)(C)C)C2 c1(C(=O)NCCNC(C2(C3CC3)CCC2)=O)cc(F)ccc1Cl c1(C(=O)NC2CC(NC(=O)CO)C2)c(Br)nc2n1CCC2 C(C(O)C(=O)NCCCCC1(NC(=O)CN2CC(C)(C)C2)CC1)=CCCC CCC(CC(=O)NCc1cc(OC)ns1)N(C(=O)CSC(F)F)C c1(C(=O)NCC2(CNC(c3nn[nH]c3Br)=O)CC2)ccc(O)cc1 C(CCCC(=O)NOCC(=O)OC)N(C(C1C(=C)C1)=O)C C(=O)(C1CCCc2nccn21)NC1(C)CN(C(c2ccn(CC(F)(F)F)n2)=O)C1 Cc1nc2cccc(C(N3C(C)C4CC3C4NC(C3(C)CCNC3=O)=O)=O)c2[nH]1 c1(OC)ccc(CNC(C)CCCC(C)C)c(Cl)c1O C=CCC(CN(CC(=O)OC)C(C1CC2CCC1C2)=O)CC(C)C C=C(Cl)CC(C(=O)NCCC(C1CCCC1)N(C)C)NC(=O)OC(C)(C)C C(C1c2ccccc2CCN1C(=O)CC1CCNC1=O)NC(c1n(C)cnc1)=O c1(C(=O)NCC(CC=C)NC(=O)C(C)Cc2ccco2)cnc2[nH]cncc1-2 c1(-n2c(-c3ncn(-c4cc(C)sc4)c3)nc(CCCN(C)C)n2)ccc(F)c(C)c1 c1(OC)cc(C(=O)NCC(O)CCNC(=O)CCC2CCC(=O)NC2)ccn1 c1(C2CN(C(C)CCC3CCCO3)C2)nc2c(s1)CCC2 C1(C(CNC(CCOC)=O)(C)O)CCCN(C(c2ccoc2CC(N)=O)=O)C1 c1(N(C(=O)C(C2CCN(C(=O)CSC(C)(C)C)C2)F)C)ccc2occc2c1 c1(C(=O)NCC2(NC(C3CC3c3ccco3)=O)CCC2)n[nH]c(C2CC2)c1Br C=CCCCCCC(=O)NC1CN(C(C2CCCCN2CCC)=O)CC1C N1(C(C(C)(CO)OC)=O)CC2(CC(NC(=O)CC3CCCCCC3)C2)C1 C1(CC(=O)N(CC(C)NC(C(C2CC(F)(F)C2)OC)=O)C)CC(=O)NC(=O)C1 Cc1nc(CC(=O)NC2CCC(CNC(c3sccc3C)=O)C2)cs1 CC1(C)COc2cc(C(=O)NC3CC(F)(CNC(=O)CCC4CC4)C3)nn2C1 C12CC3CCC1CC3NC2=O.C(CCCN(C)C)N(C)C(=O)OC(C)(C)C c1(NCC=CCC)ccc(C2CCCC(=O)N2)cc1 Cc1ncnc(C(=O)N(CCNC(=O)CCS(C)(=O)=O)Cc2ccccc2)c1C N1(C(c2cnn(CC)c2C)=O)CCCC(NC(c2ccnn2C(F)F)=O)C1C C(CCNC(C1CC2CCC2C1)=O)(C(C)C)NC(COCC)=O C1(CC)CCN(C(=O)CCOCC2CCC2)C1C(=O)NCc1c(C)coc1C N(C1CCc2cc(F)c(F)c(F)c21)CCN1C(C)CCCC1C c1(C(N2CCN(C(c3cc(CC)n(C)n3)=O)C(CC)C2)=O)c(C)cc(O)cc1O C1(C(N2CC(C)SCC2)=O)CC(C)(C)CCN1C(C1COC(=O)N1)=O C1(COC)(CNC2CC(F)(c3ccccc3)C2)CN(C(=O)C(C)CN(C)C)C1 C#Cc1ccc(CCCC(=O)NC2CCC(NC(=O)C(C)CC(F)F)C2)cc1 C(=O)(C1=CC2(CCOC2)C1)NC(C(C(=O)NCc1ccnc(C)n1)(C)C)C c1(C(CNC(C(c2cccc(Cl)c2Cl)NC)=O)=O)cc(Br)ccc1N=S(C)(C)=O CC1CC(NC(=O)C=C(C2CC2)C2CC2)CN(C(=O)Cc2cccnc2)C1 N1(C(c2cc(COC)no2)=O)CC2CCCC2(CNC(C2(F)CC2(Cl)Cl)=O)C1 Cc1oc(C)c(S(=O)(=O)NCC(O)COc2ccccc2Cl)c1C(=O)O N(C1CCCc2ccccc21)C(C1N(C(C2CNC(=O)O2)=O)CCOC1)=O O=[N+]([O-])c1cc(F)cc(S(=O)(=O)Nc2ccc(-n3cncn3)cc2)c1 c1(NC(c2ncn(C)c2)=O)cccnc1CN1CCCCC1C(N)=O c1(OCC)ccc(F)cc1NCc1ccc(F)c(OC)c1 C(=O)(C(O)CNC(C12CC(n3cc(CNS(N)(=O)=O)nn3)C1C2)=O)OC N1(C(C(C2(OC)CCOCC2)(F)F)=O)CC2(CCN2C(C2CC3CC3C2)=O)C1 c1(OC)ncc(CN(C(=O)NCC)CC2CC(C)N(C(=O)OC(C)(C)C)C2)cc1Cl N1(C(C(CC=C)C)=O)CCCN(C(=O)C2=CC(C)(C)C2)C(C)C1 n1(CC(=O)NC2CCC(NC(CC=CC=C)=O)CC2)ccc([N+](=O)[O-])n1 C(c1c(Cl)cccc1Cl)=C(C(=O)NCCC(=C)CNC(=O)C(C)CC(F)F)C C1(NC(=O)CC2C=CCC2)C2CC1CN(C(=O)CCNC(c1cccs1)=O)C2 c1(N(C(C)=O)Cc2noc(C3CC3)n2)cc(C2(C)CC2)ncn1 C1(CN(C)C(C2(C(C)(F)F)CCC2)=O)CCCN1C(C1CC2CC2C1)=O CCCCC(O)CCC(=O)NCC1(CCNC(=O)C=Cc2ccncc2C)CC1 CCC(CC)(C(=O)NC(C1CCCC1)CNC(=O)Cc1nc[nH]n1)OC Cc1cc[nH]c(=N)c1C(N1CCCC(N(C)C(C2CC2C(F)(F)F)=O)C1)=O N1(C(C2(C#N)C(C)(C)C2)=O)CCC2CN(C(c3csc(Cl)c3)=O)C2C1 C1(C)(CNC(C2C(C)(C)C2C(F)F)=O)CCN(C(=O)Cc2ccc(F)cn2)C1 C1(F)(CNC(C(CC)NC(C)=O)=O)CCCN(C(=O)C(C)(C)c2ccno2)CC1 CCC(CC(=O)N(C1CCC(NC(C2(CO)CC(F)(F)C2)=O)CC1)C)SC C1(C(N(CCCCNC(c2coc(C3CC3)n2)=O)C)=O)CC2(CCOC2)C1 N1(C(C(C#C)(C)C)=O)CC2(CCC2NC(c2nc(Cl)ccc2OCC)=O)C1 C1(CCCCNC(C2CSCCS2)=O)CCN(C(=O)C=Cc2cccnc2)CC1 CCCCC(C(=O)NCC12CC(CN1C(C1COC(=O)N1C)=O)C2)C(C)C C1(OC)CC2(C1)CN(C(=O)C(CC1CC1)NC(=O)CC(C)(C)C)C2 C1(NCc2ccc(C(=O)OC)cc2)COCCN(C(c2cc(O)ccc2I)=O)C1 N1(C(C(C)C2CC2)C(=O)NC2CCCCC2)CC2COCC2(C)C1 c1(C(N2CCCC(F)(CNC(=O)Cc3ccsn3)C2)=O)oc2ccccc2c1Cl c1(C(N(CCC(C)NC(c2cn(CC)nc2)=O)C)=O)nn(C)c(=O)cc1C N1(C(C)=O)CC2(C1)CN(C(C1CC3(CC3)CN1C(c1nonc1C)=O)=O)C2 C1(C(=O)NCC(C(=O)NCC(C)C2CCC2)O)(CO)CCCCO1 c1(CC(=O)NC(CC)CNC(=O)Cn2cc(CO)nn2)noc(C)c1C#N Cc1nc2ccccc2cc1NC(C1CC(C)CN1C(C1CC1(F)F)=O)=O C12(NC(=O)C(c3ccc(Cl)cc3Cl)O)CCC(C1)N(C(=O)CCCC1CC1)C2 c1(C(C(=O)NC2(C)CC2)N(C)CC2(OC)CCCC2)ccc2c(c1)CCC2 C1(C(=O)NC2(CN(C(CCCn3ncc(C)c3)=O)C)CC2)CC1C1CCC1 C(=O)(C1CCc2cccc(O)c21)NC(CNC(CCNC(=O)NC)=O)(C)C C1(NC(=O)NCCc2[nH]nc(C(C)C)n2)CC2CC1C1OC(C)(C)OC21 CC(C)CC(O)C(=O)NCC(C)(C1CCC1)NC(=O)C1=CCCC1C C1(C(=O)NC2CC(CNC(=O)C3=CCCOC3)C2)CCC2CCCCN12 N1(Cc2cccc(OCC)c2)CCCCC(NC(C2CC2(C)C)=O)C1 C1(C(=O)NCC(C)CCO)CCCN(C(=O)CCN(C)CCO)CC1 C=C(C)C(C)(O)C(=O)N1CCN(C(c2[nH]c(O)nc2C)=O)C(CC(F)(F)F)C1 c1(C(=O)OC(C(=O)OC)C2CCC2)c(I)cnn1C(C)C c1(NC(=O)NC(C(=O)NN2CC(C(F)(F)F)CC(C)C2)C)ccc([N+](=O)[O-])nc1 C1(CNC(C(C)OCC(C)C)=O)CC(O)CN1C(=O)C(C)c1cccs1 C=CC(C)(CC)C(=O)N1CC(CO)(NC(c2ccc(F)c(C3CC3)c2)=O)C1 N1(C(C2CCSC2)=O)CC2CCC1C1CN(C(C3CCCCO3)=O)CC21 CCCC(CCCNC(C1(c2ccccc2)CCOC1)=O)N=c1cc(C)nc(Cl)[nH]1 N1(C(CNC(Cc2c(C)cnn2C)=O)=O)CCN(C)CC1CC1OCCC1(C)C c1(N(C(C(CC#C)O)=O)C(c2cc(O)cc(=O)o2)=O)ccc2c(c1)OCO2 C1(N(C)C(c2nocc2Cl)=O)CCCCN(C(c2ccn(CC(F)(F)F)n2)=O)C1 c1(OC)ncc(F)cc1C(N1CCC(C)C(NC(=O)CC2(O)CCC2)C1)=O N1(CCNC(N2CC(=CC)C2)=O)CCCNC1=O c1(C(=O)NCC(C)(C)NC(C(C)OCC)=O)cc(S(N)(=O)=O)oc1C N1(C(=O)CCN2CCC2)CCC2CCN(C(=O)CC3CC(F)C3)C2C1 CCCC(CC)C(=O)N(CC(CC)NC(c1cc(NC(C)=O)ccc1C)=O)CC C(=O)(C(C)(F)C(=O)NCCN1CCN(C(=O)CC(C)(C)O)CC1)OC c1(CN(C2CCCC(NC(=O)OC(C)(C)C)C2)C)ccc([N+](=O)[O-])cc1 C1(O)(CN(C(c2cc(CCC)c(C)s2)=O)C)CCN(C(=O)C=CC(C)C)CC1 N1(CC)N=C(C(=O)N2CC(NC(=O)CCOc3ccc(F)c(Cl)c3)C2)CCC1=O CN1CC(O)CC1(C)C(N1CC2(CNC(C3CCC4CC34)=O)CC1CO2)=O C(c1ccc(Cl)cc1F)=CC(N1CC(CNC(c2ccc(Cl)c(O)c2)=O)C1)=O C(=O)(C(C(C)OC)NC(c1[nH]ccc1C)=O)N1C(C)(C(=O)NC)CC1 C=C(F)CN=C(NCC1CCCCN1S(C)(=O)=O)NC(C)Cc1ccccc1 c1(CC(CC)C)nc(-c2cc(OC)nn2C)n(-c2ccccc2OC)n1 N1(C(CC(C)(C)OC)=O)CCN(C(=O)CC2CCC3CC23)C(CCO)C1 CC1=C(C(=O)N2CC(F)(CNC(c3cccc(C4CCCOC4)c3)=O)C2)CCC1 Cc1cc(C(=O)NC2CCN(CCCCCSc3ccccc3)C2)co1 Cc1cncc(C(=O)NC2CCN(Cc3ccnc(O)c3)C2)c1 N1(C(C2CC(CNC(C(C)(C(C)C)OC)=O)OC2)=O)CC2(COC(=O)C2)C1 N1(C(C2CC(OC)C2)=O)CCOC(C)(CNC(C2(Cl)CC2(C)C)=O)C1 CCCCCCC(=O)NC1CC1NC(=O)C(C)(CO)OC c1(OC)ccc(C(C)C(=O)NC(C)CCN(C)C(c2ccsc2)=O)cc1OC N(C)(C(=NCc1cnnn1C)NC(CC)CC)CCOc1cccc(OC)c1 c1(C(=O)NC2(C(=O)NCC3(OC)CCC3)CSC2)cn(C)cc1C C(N=c1cc[nH]cc1[N+](=O)[O-])C1(CC(N2CCOCC2)=O)CCCC1 C1(NC(CC(=O)NCC)=O)C2CCC(C2)C1C(=O)N(CC(C)(O)C1CC1)C CC1CCN(C(=O)C(c2ccn(C)c2)C)C1C(=O)NCC1CNC(=O)CO1 C(=O)(C(C)C(C)(C)C)NC1CCC(N(C(COCCC)=O)C)CC1 N1(C(COCC(=C)C)=O)C2CCC1CN(C(C1(OC(C)=O)CC1)=O)C2 CC(C)(O)CCC(=O)NCC1=CCN(C(C2CSCC(=O)N2)=O)CC1 N1(C(c2c(C(=O)OC)coc2)=O)CCCN(C(c2ccc(C(F)(F)F)o2)=O)CC1 N1(C(c2c(C)nsc2)=O)CCN(C(c2cncc(F)c2C)=O)CC1CC(F)F CC1CN(C(C2CCCC(O)C2)=O)CC1CNC(C1CC(N(C)C)C1)=O C1(c2ccccc2)(NC(=O)C(O)C2CCC2)CN(C(c2nc(C3CC3)cs2)=O)C1 c1(C(N2CCN(CC(N3CC(C)OC(C)C3)=O)CC2)=O)cn2ccccc2n1 Cc1cccc(C(=O)NCC2(CC(=O)NC(C)C(=O)NC(C)(C)C)CC2)c1O N1(C(CS(CC)=O)=O)CCC(C)C(CNC(=O)C(C)(C)c2nccs2)C1 c1(CC(=O)NC(C2CC2(F)F)CC)ccc(S(C)(=O)=O)c(C)c1 C12(CC)CCC(C(N3CCCC(CNC(c4cnccc4C)=O)C3)=O)(CC1)CO2 c1(NCC2C(C)(C)C2CO)cc(=NC2CCc3c(Cl)cccc32)[nH]c(C(F)(F)F)n1 c1(C(N2C(CNC(=O)CC3CN4CCN3CC4)C=CC2)=O)ccnc2ccsc12 C1(N(C(CC)CNC(c2nocc2C(C)C)=O)C(C2CCCC2)=O)CCC(C)CC1 N1(C(CSCC(=O)OC)=O)CC2CCCC(N(C(=O)C(C3CC3)C3CC3)C)C2C1 c1(CC(=O)NCC(F)CNC(C2CC3CCC2CC3)=O)cccc2cnccc12 c1(CC(=O)N(CC(C)NC(C2CC2(F)F)=O)C)nc2ccccc2s1 N1(C(CC(=C)Br)=O)CCN(C(c2ccc(N)c(O)c2)=O)CCC1C CCC(F)(F)C(C)(C)C(=O)N1CC2(CNC(=O)CC(C)F)CC1CO2 c1(C(=O)NCC=CCNC(C=CCCC)=O)cccc(OC)c1 c1(OC)cccnc1CCC(=O)NCCC1CSCCN1C(C1CCC(O)CC1)=O N1(C(c2nc(C#C)sc2)=O)CC2(C1)CN(C(=O)C(O)CC(N)=O)CC2CO C(=O)(CC(C(F)F)C(C)(C)C)NC(C(C)C)CNC(c1nsnc1O)=O C1(C(=O)NCC2N(C(CNC(CC)=O)=O)CC2)CCCN(c2cc(C)ncn2)C1 C(=O)(CC(C)(C)C(C)(F)F)NCC1C(C)CCN1C(C1CCCC(O)C1)=O C(=O)(C(C)C(O)C(C)CC)NCC1(C(N2CCC(OCC(C)C)C2)=O)CC(=C)C1 C1(CNC(=O)NC2CCC(NC(C)=O)CC2)CC2(C1)CC(F)C2 c1(SC)nc(O)c(C(=O)OC(c2ccc(F)cc2Cl)C)cc1C#N CC1=C(C(=O)NC2CCN(C(=O)Cc3ccc(Cl)s3)CC23CCC3)CCS1(=O)=O c1(C(=O)NC(C(=O)NCC2C(OCC)CC2)C2CC2)cnc(Cl)s1 Cc1cc(C)n2ncc(C(N3CCC4(CC(NC(=O)C5=CCC5)CO4)C3)=O)c2n1 c1(C(N2CC(F)CC2c2nc[nH]n2)C(=O)NCC(=C)C)oc2ccccc2c1Br C(=O)(C1=NOC2(CCOC2)C1)Nc1cccc(NC(C(F)OC)=O)c1 c1(NC(C)Cc2ccco2)ccc(S(=O)(=O)NCCC2CCCN(C)C2)cc1Br Cc1ccc(OC(N2CCCC(NC(C)(C)C)C2)=O)cc1[N+](=O)[O-] c1(C(=O)NCC2CCCN(C(C3(C)C=CCC3)=O)C2)ccnc(Cl)c1O Cc1cc(COCC(=O)NCC2(F)CN(C(C34CCCC3C4)=O)C2)no1 c1(-n2cc(-c3c(C)con3)nn2)cccc(CCNC(C2CCS(=O)(=O)N2)=O)c1 S(=O)(=O)(CC(=O)N1CCCC1CCNC(C1CC(n2cnnc2)C1)=O)NC C(C(C)(C)C(C)(F)F)(c1nnnn1C(C)(C)C)NCCc1ccnc(C)n1 c1(CC)nn(C)cc1C(=O)NC1CC(F)(CNC(=O)CCn2ccccc2=O)C1 C1(CC)CN(C(c2csc(-c3sccc3Br)n2)=O)CCC1CC(N)=O N1(C(C(CC)N(C(=O)CCc2ccsc2)C)=O)CC(C)C(O)C(C)C1 c1(Cn2c(CN(CC(=C)C)CC3CCCO3)nnn2)cccc2ccncc12 C1(CNC(c2nc(CC)sc2)=O)CC2CCC1N2C(=O)CN1CCC1 O=C(C1=COCCC1)NC1CCN(C(c2ccc(Br)c(F)c2)=O)C1C1CC1 c1(CCNC(N2CC(CN(CC)CC)C2)=O)ccccc1SC(F)(F)F C1(N(C(CSSC)=O)CC)CCCN(C(C2CCCN(CC(F)F)C2)=O)CC1 C(=O)(CC(C(C)CC)NC(=O)C(C)(O)CCN(C)C)NCC1N(CCC)CCC1 C(=O)(CCCCCn1cc(CCC(C)O)nn1)NC1(COC)CCCC1 N1(C(c2c(CC)ccs2)=O)CC(NC(=O)C2=CCCSC2)CC1(C)C C1(C)(C(=O)NC(COCC)(C)C)CCCN(C(c2cccc(F)c2)=O)C1 C1(C(=O)NCC2C=CC(NC(CC)=O)C2)C2C=CC(CC2)C1C(=O)NC O=Cc1cccc(CN2CCOC(C(=O)NCCc3cccc(F)c3)C2)c1Br C1(N(C(CCc2c(C)ncs2)=O)C)CN(C(=O)CN2C(=O)CCC2=O)CCC1O N1(C(c2cc(CSC)c(C)s2)=O)CC2CCN(C(=O)C(C)c3cncs3)CC2C1 c1(C(=O)NCC(CNC(C2(Cl)CC2(C)C)=O)OC)ccn2nccc2n1 c1(OC)ncccc1C(N1CCOC(CCCNC(c2coc(OC)n2)=O)C1)=O c1(CN(C(CCC#C)c2ccccc2)C=O)cc(C)ccc1Br N1(C(CCC#C)=O)CC2CCCC(NC(c3ccc(=O)oc3)=O)(C2)C1 C1(NC(COCCCOC)=O)CN(C(c2c(C)cnnc2O)=O)CCC1O C(=O)(C(C)(C)C1CCOC1)N(CC(=O)NC1CC(CC)C1)C1CCC1 O=[N+]([O-])c1nn(-c2ccc(F)cc2)nc1Sc1cccnc1 C12(CNC(c3n(C)nc(O)c3)=O)CN(C(=O)CNC=O)CC(F)(C1)C2 n1(CC(=O)N(C(C)CNC(=O)C(=Cc2cccs2)C)CC)ccnc1C C(=O)(C(C(C)CC(C)(C)C)N1CCOC(C)(c2cccc(Br)c2)C1)NCCSC C1(N(C(=O)CC2CC=CCC2)CC)CCCN(C(=O)Cc2nonc2C)C1 C1(CC(N2CC(C(=O)OC)(COC)C2)=O)CCCN(C(=O)CSS(C)(=O)=O)C1 c1(C(=O)NCC(C)NC(C2CC2c2ccco2)=O)nc(Br)sc1Cl c1(C(=O)NCC2CC(NC(C3N(CCC)CCC3)=O)C2)cnc(O)c(Br)c1 c1(CC(=O)N(CC(C)NC(=O)CNS(C)(=O)=O)CC)occc1C C(CN=c1[nH]c(=NCC(C)N2CCC(C)CC2)c2ccc(OC)cc2[nH]1)OC N1(C(CCC(C)N(C)C)=O)CCOC2(CCC(NC(c3cn(C)cn3)=O)CC2)C1 C(CN=c1nc2sccc2c(NCC2CCCC2(F)F)[nH]1)(C1CCC1)OCC Cc1nc(C(N2CC3CC(NC(=O)CCC(C)(F)F)C(C3)C2)=O)c(=O)[nH]c1C CC1(C)COC(CC2(C(=O)NC(c3ccc(F)cc3)CCO)CC2)C1 Cc1ccccc1-n1nnnc1C(C)C(=O)NCCCN(c1ccc(Cl)cn1)C c1(CC)csc(C(c2nnnn2C(C)C(=O)OC)NCCOC(C)C)n1 c1(C(N(CCNC(C2CCC(=O)N2)=O)CC)=O)ncc(F)cc1C C1(O)(CNC(C2C(NC(C3(CC)COC3)=O)CCCC2)=O)CCCCCC1 N1(C(c2cnn(C3CC3(F)F)c2)=O)C2CCC1CN(C(C1(CF)COC1)=O)C2 C1(C(C)(C)NC(C2C(C)C2)=O)CCCN1C(c1ccoc1C(F)(F)F)=O C(=O)(C(C)(F)C(F)(F)F)NCC1CC(OC)CN1C(=O)C=Cc1ccncc1 Cc1ccc(C)c(N(C)C(C2CCN(C(c3cnc(C)nc3C)=O)C2)=O)c1 C1(NC(c2nc(CC)oc2C)=O)CCN(C(=O)C(O)C(C)(C)C)C(C)C1 N1(C(c2cc(OC)n(C)n2)=O)CC2CCC1C1CN(Cc3nonc3C)CC21 C(CC(C(=O)NC1CC(n2ccnn2)C1)NC(c1cc(Cl)n[nH]1)=O)SC c1(NC(C2CN(C(C3CCN(C)CC3)=O)CC(F)C2)=O)cc(F)c(Cl)nc1Cl C1(C(C)=O)CC(C(N2CC(NC(c3ccns3)=O)CC2C)=O)C1(C)C c1(SCCC)ccc(C(=O)NCC(C2CC2)NC(c2cn(C)nc2CC)=O)cc1 c1(SC)cccc(CC(=O)NC2CC(CCNC(=O)CSc3ccncc3)C2)c1 c1(C(=O)NC(CN(C(=O)C(C)CC2CCCCC2)CC)C)c[nH]c(=N)o1 C1(n2cc(CNC(CC)=O)nn2)CCCN(C(=O)C(C)CN(C)C(C)=O)CC1 N1(C(C2(C)CNC(=O)N2)=O)CCC2(CC1)CC2C(=O)NCCCn1cncn1 C1(CC)(CO)CCCN(C(=O)C(O)C2CN(C(C34CCC(CC3)CO4)=O)C2)C1 CCC(CCC(=O)Nc1ccc(O)cc1CO)NC(=O)Cc1cncs1 C(CN=[N+]=[N-])(C(=O)NCC1(C)CNC(=O)O1)NC(c1ccc(C(C)=O)o1)=O CCC(CC(C)C)C(=O)NC1CN(C(=O)Cc2cccn2C)C1 C1(CNC(C)=O)CCN(c2nnc(CC3CCCC3)n2CCCS(C)(=O)=O)CC1 Cc1cc(C(F)(F)F)ncc1C(N1CC(CC(C)NC(c2cccn2C)=O)C1)=O c1(OC(C(=O)NCC(CC)NC(C2(CO)COC2)=O)CC)cccc(Cl)c1Cl C1(NC(=O)CONC(c2n[nH]c(O)n2)=O)C(=O)OC2CCCC12 Cc1ncnc(C(N2CCC(CCCNC(=O)C(O)P(C)(C)=O)CC2)=O)c1C C(=O)(CC(O)C(C)(C)C)N1C(CCNC(CC)=O)CCCC1 c1(CNC(C=CC2(C)COC2)=O)nnc2n1CCN(C(c1ccc(CO)o1)=O)C2 c1(C(=O)OC)sc(C(N2CC(O)CC2CNC(=O)C(F)n2ccnc2)=O)cc1C C(=O)(C#CC1CCCCO1)NC1(C2CN(C(C(CC)C(C)C)=O)C2)CC1 Cc1cccc(C(=O)N(CCCNC(=O)CCc2nnc(C(F)F)o2)C2CC2)n1 CCCCCC(C)CC(=O)N1CCN(C(C2CC(C)(F)C2)=O)C(C2CCCC2)C1 N1(C(C2(OCC)CCCCC2)=O)CCCC(COC)(NC(=O)C=C(C)Cl)C1 C1(C(=O)NCCCN(C(c2cc(C)n(C(F)F)n2)=O)CC)COC(=O)N1C c1(C(C(=O)NC(CC(C)NC(CC=CC=C)=O)C)C)nc(F)ccc1Cl C1(NC(CSCCOC)=O)CCC2(CCN(C(C3Cc4cccnc4C3)=O)C2)C1 c1(C(C)NCc2ccc(OCCc3ccccc3)cc2)nnc2n1CCOC2 Cc1cc(N2CC(C)C(C)C2)ncc1S(=O)(=O)N1CCC(CCCO)CC1.NC c1(C(C)C)nccc(C(=O)NCCC2CSCCN2C(C2CCCC2O)=O)n1 C(=O)(C(C(C)(C)C)C1CCCO1)N1CCC(OC)(CNC(C2CC(O)C2)=O)C1 N1(C(c2n[nH]c(C)c2C)=O)CCN(C(c2cnn(C3COC3)c2)=O)C(C)C1C N#Cc1nc(=NC2C3CC2CN(C(c2cc(-c4cccs4)on2)=O)C3)cc[nH]1 C(=O)(CC(C)(O)C(F)(F)F)NCC(CNC(c1n(C(C)C)ncn1)=O)(C)O c1(C(N2CC(Cn3cc(C4(C)CCCC4)nn3)OCC2)=O)nccn2ccnc12 Cc1onc(CO)c1C(N1CC(NC(=O)CCCC#N)C(c2ccnn2C)C1)=O Cc1ccc(C(=O)NCC2CCCN2C(C2CC(=C(F)F)C2)=O)cc1O c1(C(N2C(C(C)NC(CCOCC(C)C)=O)CCCC2)=O)c[nH]c2ccncc12 Cc1cc(C(=O)NCc2cc(C(=O)NC(C3CCCO3)CO)co2)ncc1N c1(C(N(C(CCNC(c2cc(C)sc2C)=O)C)C)=O)cc(Cl)ccc1F CCC(C)(C(=O)NCC1CC(F)CN1C(c1cc(CN(C)C)c[nH]1)=O)C(F)F C#CCCCC(=O)N1CCOCC1CCNC(c1sc(NC2CC2)nc1C)=O Cc1nn(C)cc1S(=O)(=O)N(C)CC1CCN(C(c2ccc(F)nc2)=O)C1 c1(C(=O)NC2(C)CC(NC(C3CN(CC(C)C)C(=O)C3)=O)C2)ccn2ccsc12 N1(C(c2cc(C)c(C)s2)=O)CC2CCC1CC2NC(C1(F)CCCC1)=O Cc1c(C(F)(F)F)n[nH]c1C(=O)NC(Cc1cn[nH]c1)C(=O)N(C)C CC1CC(C(=O)NCC(O)CCC2CC2)N1C(=O)COC1(C)CCC1 C1(CNC(=O)C=C(Cl)Cl)CN(C(=O)COc2cccc(F)c2)CCC1(F)F C(=O)(C(O)CC(N)=O)NC(C(C)C)CCN(C(=O)Cc1cnc(C2CC2)[nH]1)C N1(C(CC2CC(=O)NC2=O)=O)CC2CC1CN2C(c1ccccc1)=O c1(CC)nc(=NCC(C)NC(c2ccc(-n3cncn3)nc2)=O)s[nH]1 CCCC(C)CC(=O)NCCCC(C)NC(=O)Cc1c(C)nn(CC)c1C C1(NC(CC(=O)NCC#C)=O)CN(C(C2CCCN(C(C)=O)C2)=O)CCC1O c1(C(=O)NCC2C(NC(CCc3n(C)cnc3)=O)COC2)scc2c1CCCC2 C1(CC(=O)NC(c2ccccc2Cl)COC)CCC2(CCC2)CO1 C=C(C)CCCC(=O)NC1(C)CCN(C(=O)C(C)N=[N+]=[N-])C1 c1(CC)nn(C)cc1C(=O)NC(C)CCN(C(=O)C(C1CCCN(C)C1)(C)C)C C(=O)(CS(=O)(=O)CCOC)NC1CN(C(C23CC(CC)(C2)C3)=O)C(CC)(CC)C1 N1(C(CC=C)=O)CC(NC(c2cnc(C(F)F)nc2)=O)CC1C c1(CN(C(C)Cc2ccc(OC)cc2)CC)cncc(C(C)(C)C)c1 C(=O)(CCC(=O)c1cccnc1)NC(C)(CNC(=O)C=Cc1ncc[nH]1)CO c1(CC(C)C)ccccc1C=O.c1(SCC(=O)OC)nnnn1C Cc1cnc(NC2CN(C3CCOCC3)C2)c(S(=O)(=O)N2C(C)CCC2C)c1 Cc1cnc(C(=O)Nc2cccc(NC(c3ccn(C)c3)=O)c2)nc1 N1(C(c2n(CC)ccn2)=O)CC(NC(C2CCCC(C)C2)=O)C2(CCOCC2)C1 c1(C(N2C(CC(=O)N(CCC)C(C)=O)C(=O)NCC2)=O)cnn2c1OCC(O)C2 C1(C)(CNC(CCN2CCN(C)CC2)=O)CCCN(C(c2cc(C#N)on2)=O)C1 c1(C(N(c2cccc(C(=O)O)c2)C)=O)cccc(OCCS(C)=O)c1 c1(C(=O)NCC(CNC(=O)C=C(C)C)OC)cc(N)ccc1C c1(CC(=O)NC2C(NC(c3c(C)cno3)=O)CCOC2)cnc2n1CCOC2 C12(C(N(CCCCC=C)C)=O)CC(CO1)N(C(C1CCOCC1)=O)C2 C1(C(N(CC(C)N(C(C)=O)C)C)=O)(NC(=O)CC2CCSC2)CCN(C)C1 N1(C(C(C)C2CC2)=O)CCC(C)(C)C1C(=O)NCC1CCCCC1(C)C CCC(C)C(C)C(=O)NCCCN(c1nc(Cl)ncc1C(N)=O)C C(CC(CO)N=c1cc(F)nc(C(C)(C)C)[nH]1)N(C)C c1(C(N(CC(=O)N(C)CC)CC#C)=O)ccc(F)nc1 C123CC(CN1C2)C3.C1(CNC(N(C)Cc2ccccc2)=O)CCCC(N)C1 C(=O)(C(CC(C)C)N(C)C(C1CN(C(C)C)C1)=O)N1CCC(C(CC)C)CC1 c1(C(=O)NCCC(C)NC(c2cc(-c3ccoc3)[nH]n2)=O)cnc(N)c(N)c1 C1(CC)CCCN(C(c2nn(C)cc2C(N2CC3C(C2)C3(F)F)=O)=O)C1OC C=CC(CC)CC(=O)NCC1COCC1NC(=O)CN1CCC(C(N)=O)CC1 c1(C(=O)NC(C(C)C)C2CCC2)n[nH]c2c1CN(C(c1c[nH]nc1C(C)C)=O)C2 N1(C(C(C)=CC)=O)CC(OC)C(OC)C1CNC(=O)CC(C1CC=C(C)CC1)C C1(C(C)NC(=O)C(c2ccc(C)cc2)O)CCN(C(c2cnc(S)nc2)=O)CC1 CC(CCC(C)(C)C)C(=O)NCCOCCCNC(c1cncc(C(F)F)c1)=O C(C1=NOC2CCCCC12)n1cc(CCCNC(c2cccc(Br)c2F)=O)nn1 c1(C(N(CCC(C)NC(c2ccc(C3CCCO3)[nH]2)=O)C)=O)csc(=N)[nH]1 c1(C(N2C(CCNC(CN(CC)CC)=O)COCC2)=O)csc2nccn12 CCC(C)(C)C(=O)N(C(CNC(=O)CC1CCCC12CC2)C1CC1)C C(CCCC(CO)NC(=O)CC(C)CF)NC(c1c(C)c[nH]c1)=O N1(C(C(CC)C#N)=O)CCCC2(NC(C3CC4CC4C3)=O)CCCC12 c1(C2CCN(C(C3N(CC)CC3)=O)C2)ccc(NC(=O)CCNS(C)(=O)=O)cc1 C12(C(=O)NC3C(NC(CC4CN(C)C4)=O)COC3)CCC(=O)N1CCS2 C1(C(=O)NCCN(CCC)CC)(CNC(=O)Cc2cc(C)cs2)CCCO1 N1(C(c2cn(CC(C)C)nc2)=O)CCC(CN(C(=O)C=C2CC2)C)CC1 C#CCC(C(=O)OC1CC(OCC2CC2)C1)NC(=O)C(C)OCC c1(C(C(=O)NCC2COCCN2C(c2cnn[nH]2)=O)O)ccc(Cl)cc1F Cc1ncsc1COCC(=O)NCCCCCN(C)C(c1n[nH]cc1C(C)C)=O C1(C)(CNC(c2ccc(C)cc2)=O)CCCN(C(=O)CC2CSC2)C1 CC1=CCC(C(=O)NCC2CCN(C(=O)C(C)(C)c3cccs3)CC2)CC1 C(=O)(C1COc2ccc(Cl)cc21)NC1C2OCC(NC(=O)CCC(F)F)C2OC1 Cc1cc(N2CCC(c3cc(F)ccc3Cl)CC2)nc(N(C)CCOC2CC2)n1 c1(OC)cc(C)c(C(N2CCC(CF)(NC(=O)CN=S(C)(C)=O)C2)=O)cn1 CCS(=O)(=O)C=CC(=O)NCC1CCCN(C(c2csc(C#N)c2)=O)C1 N1(C(Cc2nc(CC)sc2)=O)CCC(C2CN(C(=O)C(F)n3ccnc3)C2)CC1 C(=O)(C1=CCCCCC1)N1C(CC(=O)NCc2n(C(C)C)ncc2)CCC1 C1(NC(C(C)(N(C(C(CC)OCC)=O)C)C2CC2)=O)CC(CO)C2CC12 CC(c1cccnc1)=CC(=O)NC(C)CNC(=O)C(c1ccc(N(C)C)cc1)C N1(C(C(C)(C)O)=O)CC2CCCC(CNC(C3CC34CCOCC4)=O)C2C1 C(=O)(CCCCN=[N+]=[N-])N1CCC(C(=O)NC2(C(=O)OC)CC2C)CC1 C(=O)(C(F)CC(C)(C)C)N1CCSCC(C)C1.C1(=O)C(CC(F)F)N1 C12(C(C)C)COC(C(=O)NCC3CCCCC3CNC(=O)Cc3cc[nH]n3)(C1)C2 c1(C(=O)NCC2CN(C(c3nn[nH]c3C(F)(F)F)=O)CCO2)cc(Cl)c(Cl)nc1Cl C=CC(C)(O)CCCC(C)C(=O)N1CCC(CCNC(=O)C(F)=CC2CC2)CC1 C1(N(C(C(CC)SC)=O)C)CC2CCC(C1)N2C(=O)Cc1ccc(C)nc1 c1(C(=O)NCC2C3CN(C(C4(C)CC4(F)F)=O)CC32)[nH]nc2ncnc(O)c12 C(CNC(=O)Cc1nocc1C)(CC(=O)N(C)Cc1csc(C)n1)OC CC1C(C=CC(=O)NCCCOCCNC(C2(C)CCCOC2)=O)C1(Cl)Cl N1(C(c2ncn(C)c2)=O)CC2(CCN(C(=O)C(c3ccc(Cl)cc3F)O)CC2)C1 N1(C(C=C(C)Cl)=O)CC2CCN(C(=O)CCOc3ccccc3)C2C1 Cc1sc(=NC2CCOC(C(C)(C)C)C2)[nH]c1-c1cccc(F)c1 N1(C(C(CC#C)C2CC2)=O)CCN(C(c2cc3occc3[nH]2)=O)CC1C1CCC1 c1(C(=O)NC2C(CNC(C(CSC)C)=O)CCCC2)ncnc2c1cnn2C Cc1cn2c(n1)C(C(=O)N1C3CCC1CC(NC(C1CC(CF)C1)=O)C3)CCC2 c1(CCNC(CC)(C(=O)N(C)C)c2ccccc2)ccc(SC(C)C)nc1C C1(OC)CC(CNC(=O)CC2(C)CCOCC2)N(C(c2cnc(Br)s2)=O)C1 Cc1cc(C(=O)NCC2(O)CCN(C(=O)C=Cc3cn(C)cn3)C2)c(C)s1 c1(C(=O)NC2CCN(C(CCCOCC=C)=O)CC2F)nnc2n1CCCC2 C1(CC(=O)NCC2(OC)CN(C(Cc3ccc(OC)s3)=O)C2)COCC(C)(C)O1 c1(C(=O)NC2C(NC(CC=CC=C)=O)C2)cc(N2CCNC2=O)ccc1F Cc1ccc(=O)n(CC(N2CCCC(N(C)C(c3ccncc3Br)=O)C2)=O)c1 c1(C(C)N)cccc(OCC(=O)NC(c2ccccc2)c2cccs2)c1 C(=O)(CS(=O)(=O)CC(F)(F)F)N1CCC(N(C2(Br)CC2)C(C)(C)C)(CNC(C)=O)CC1 Cc1nc2[nH]c(C(=O)N(C(C)CNC(=O)COCC3CCC3)C)cc2s1 N1(C(C2C(C)(C)C2)=O)CC(CNC(=O)CNc2ccccc2C(F)F)CC1(C)C CCCC(C(=O)N1CCN(C(c2c[nH]c(C#N)c2C)=O)CC1CC(F)F)C(C)C Cc1sc(C(=O)NC(C2CCN(C(=O)COC(C)C)C2)C)cc1Br C(=O)(C(=O)C(C)C)N1CC(CC(=O)N(CC(F)F)CCO)(OC)C1 CC1CN(C(c2nc(Cl)cs2)=O)CC1NC(C1(c2cccnc2)CCC1)=O N12CC3(CCC3)CC1C2=O.c1(CC)c[nH]cc1C(N1CCC(C(C)(C)OC)C1)=O N1(C(CCCCC=C)=O)CCC2(CCCN(C(=O)CC3CCCN3C(C)=O)C2)C1 C1(CC)CCCN(CC(=O)NCC2(CN(C)C(C3C(Cl)(Cl)C34CC4)=O)CC2)C1 N1(C(c2c(CC)scc2)=O)CCCN(C(C2CCC(O)CC2)=O)CC1C S(=O)(=O)(c1ccc(N2CCC=C(C)C2)c(F)c1)NC(c1ccncc1)CC CCC1=C(C(=O)NCC2=CCN(C(c3cccc4cc[nH]c34)=O)CC2)CCCO1 c1(C(=O)NCC(CN(C(C(C)SCC)=O)C)O)ccc(Cl)cc1Br C1(NC(CC2CC(C)C2)=O)CCCN(C(c2ccsc2)=O)C1C C1(F)(C(=O)NCC2CCN(C(c3ncsc3C(F)(F)F)=O)CC2)CCCCCC1 c1(C(N2CCN(C(CCNC(=O)NC)=O)CC2CF)=O)nn(C)c2ccccc12 N1(CC(=O)NC(C2CN(C(c3scc(C(=O)OC)c3)=O)C2)C)C(=O)CN(C)C1=O Cc1oncc1S(=O)(=O)N1CC(CC(N2CCC(C(c3nccs3)=O)CC2)=O)C1 C12(C(=O)Nc3cccc(-c4ccc(CC)cc4)c3)C3C4C1C1C2C3C41CO c1(OC)cc(O)c(C(=O)NCC2CCN2C(=O)C(C)(C)NC(C)=O)cc1Br c1(CNC(C2(C(F)F)CCNCC2)=O)cnn2ccccc12 c1(C(N(CCOC)CCNC(=O)Cc2csc(C)c2)=O)ccc(Br)cn1 c1(CN2CCC(NC(c3ccc(C(=O)OC)cc3C)=O)C2)ccc2cc[nH]c2n1 c1(C(=O)NC(C(=O)NCC2(CO)C(C)(C)C2)C2CCCC2)ccc(=N)[nH]c1 CCCC(CCCNC(c1cnc(O)cc1C)=O)NC(=O)Cc1c[nH]nc1O c1(CC)n[nH]cc1C(=O)NC1CC1NC(c1coc(C2CCCCC2)n1)=O C1(S(C)(=O)=O)(C(=O)NC(CNC(c2cn(C(C)C)nc2)=O)C(C)C)COC(=O)C1 N1(C(Cc2cnc(C)s2)=O)CCC(F)(C(=O)NCC2(O)CCCOC2)C1 C(=O)(CC(O)C(C)C)NCCN(C1CCCCC1)C(c1c(C#C)c[nH]n1)=O c1(C(NNC(COc2cccc(SC)c2)=O)=O)ccc2c(c1)OCO2 Cc1ccc2sc(C(N3CCN(C(=O)C=Cc4scnc4C)CC3)=O)cc2c1 c1(C(N2CCN(C(C3CCCCCC3)=O)C3CC23)=O)cc2cccc(Cl)c2[nH]1 C1(OCC)CC2CN(C(=O)C(C3CC3)N(C(=O)C(C)C(C)NC(C)=O)C)CC12 C(C)(CC(F)(F)F)NC(CCCNC(C1(OC)CCSC1)=O)=O C1(C)(NC(c2n(CC)ccn2)=O)CCCN(C(c2ccc(OC)c(N)n2)=O)C1 C1(CNC(C2CCCSC2)=O)CC2CC2N1C(c1cnc(OCC(F)F)cn1)=O C=C(C)CC(C)C(=O)N1CCC(C(C)NC(c2cscc2SC)=O)C1 Cc1nc([N+](=O)[O-])cn1CC(N1CC2C(N(C)C(C3CC(F)CN3C)=O)C2C1)=O C1(CNC(C(C)S(C)(=O)=O)=O)CC12CCN(C(=O)C=CC1CCCC1)CC2 C1(N(C(=O)CCCc2cccs2)C)CCC(NC(C2CCC2(F)F)=O)CC1 C(=O)(CCCCN(C)C)NCCN(C(c1ccc(C(=O)OC)o1)=O)CC C1(C(=O)NCc2cccc(CNC(CCC(C)C)=O)c2)OCC2CCCCC12 c1(NC(C2(COC)N(C(CCCC)=O)CC=C2)=O)ccc(C2CC2)nc1C c1(N(CCN(C(=O)CCc2cccs2)C)C)cccnc1C(F)F CCC(N=c1ccnc(NCc2ccccc2-c2cccnc2)[nH]1)C1CCCO1 c1(NC(C)=O)cc(Br)ccc1C(=O)Nc1cccnc1C(=O)N(CC(F)F)C C(C(C)(C)C#CC(=O)NC(CCO)c1ccco1)NC(C1CCN(C)C1=O)=O c1(C(N(C)CC2COCCN2C(C2COCCO2)=O)=O)cc2cn[nH]c2cn1 C1(C(=O)NCC2(CO)CCCO2)CCCCC1NC(C1CCCC1O)=O c1(C(N2CCCCC(NC(C3(C(C)C)CC3)=O)C2)=O)cc(F)c(F)c(F)c1 c1(C(=O)NCCC(=O)Nc2cccc(C3CC3)c2)cn2c(n1)CCC2 N(C1CCc2ccc(Cl)cc21)C(C1COCCN(S(CCC(=O)OC)(=O)=O)C1)=O N1(C(c2cc(C)n(C(F)F)n2)=O)CC(NC(c2cccc(Cl)c2N)=O)CC(O)C1 c1(CC)onc(C)c1NC(c1ccn(CCNC(=O)CCN(C)C)c1)=O C12(CNC(c3c(Cl)cccc3Cl)=O)CCC(CC1)CN2C(=O)Cc1cnccn1 CC1=NOC2(C1)CC(C(=O)NCCN(C(c1cc(F)c(Cl)cc1F)=O)C(C)C)C2 C(=O)(C(O)CC(F)F)N(C)C(c1ccc(Cl)cc1)c1ncc[nH]1 C1(O)(CNC(C2(CC)CCC2)=O)CCCN(C(C2CN(C)C(=O)CCO2)=O)CC1 c1(CN2CC3(CC(NC(C4(F)CCCNC4)=O)C3)C2)cc(F)c(F)cc1Cl C1(C(N(C2C(C)CCC2)C)=O)CC(O)CN1C(C1CC(F)C1)=O N1(C(C2CCC(C)CC2)=O)CCCC12CCN(C(=O)C(F)CC1CCOC1)C2 C1(C(N(CCCCCNC(=O)CCC2CCCO2)C(C)C)=O)C2CCC3C(C2)CC13 c1(C(=O)NCc2cc(C(N3C(COC)CCCC3)=O)ncc2)cnccc1C#N C1(C(=O)NC23CC(CNC(C(C)OCCOC)=O)(OC2)C3)CCOCC12CCC2 N1(C(c2cc(C)ns2)=O)CCCC12CCN(C(=O)Cc1ccc(F)cn1)CC2 C=CC(CCC)CC(=O)NC1(C(N2CC(O)(CCC)C2)=O)CC1(C)C C1(C)(CNC(C2(CCNC(CNC(CN(C)C)=O)=O)CC2)=O)CCCO1 C1(C(=O)NC)CCN(C(C2(C)CN(C(=O)CNC=O)C2)=O)C1 c1(CCC(=O)NC2CCC2CNC(=O)Cc2ncoc2C2CC2)ccc(Cl)s1 N1(C(c2c(C)csc2)=O)CCCN(C(C2CCCC(C(N)=O)C2)=O)CCC1 C12(CC)CC1CN(C(c1cc(O)n(C)n1)=O)C2 C(=O)(C(=O)C(C)(C)C)NC1(C(=O)NC(c2cnccn2)C)CC(F)C1 c1(OC)cccc2cc(CNCC(C)(C(=O)O)n3cc(Br)cn3)oc12 N1(C(C2N(CC)CCC2)=O)CC(F)(F)CC1CNC(C1CCCN1)=O C(=O)(C1=CCCOC1)NCC(=O)NCC12CC(CN1C1CC1)C2 c1(CC(=O)NC2CCCC(N(C(=O)CC3CC3)C)C2)cccc(C#N)c1 C(C)(CC(=O)NCCCCN(C)C1CC1)NC(C(N1CCNC1=O)C)=O c1(NC(C2CC3CC3N2C(c2ccc(O)nc2)=O)=O)cccc([N+](=O)[O-])c1Br C1(CC(=O)NC(CC=C)CNC(c2ccc(Cl)cc2N)=O)COCC(C)(C)O1 c1(C(=O)NC2CCC(Cn3cc(CSCC)nn3)CC2)cccn2c(C)cnc12 c1(C(=O)NC2C(CNC(CCCOC(C)C)=O)CC2)cn2c(n1)SCC2 Cc1ccc(O)cc1C(N1CCC(C(C)CNC(=O)CO)CC1)=O c1(C(=O)NC(C2CCN(C(CC3C(C)OCC3)=O)C2)C)cnn(C)c1C(F)F Cn1nc(C(F)(F)F)cc1NCC1CCC(C(=O)NCc2ncccn2)CC1 c1(C(=O)NC(C2CCN(C3CCN(C)C3=O)CC2)C)cc(F)cc(F)c1 C1(NC(CC(C=C)C)=O)CCC2(CCN(C(C3CC(C)CCO3)=O)C2)C1 C1(C(N2CC(CN(C(Cc3c(C)n(C)nc3)=O)C)OCC2)=O)CC12CCSCC2 N1(C(C(c2ccc(Cl)cc2)C)=O)CCC2(CC1)OCCC2NC(=O)CC(F)(F)F c1(NCC(C)NC(=O)OC(C)(C)C)cc(N(C)CC2CCCCN2C)ncn1 C1Cc2ccc(Br)cc2C1.c1(C(C)(C)NC(=O)N)cc(O)n[nH]1 N1(C(c2c(C)ccs2)=O)CCN(C(=O)Cc2ccc3c(c2)OCO3)CC(CO)C1 c1(-c2nc(NC(C(C)NC(c3ccccc3)=O)=O)sc2)ccc([N+](=O)[O-])cc1F Cc1c(C(N2CCN(C(C3(C(=O)C4CC4)CC3)=O)CC2CCO)=O)cncc1Cl C12(NC(COC)=O)CC1CN(C(=O)C(C)Cn1cccn1)C2 C1(C(C)NC(C=COCC)=O)CCCN(C(c2cc(C(C)(C)C)[nH]c2C)=O)C1 C(CN=c1[nH]c(C2CC2)nc(Cl)c1C)OCCN(C(C1C(OC)CC1)=O)C N1(C(C2C3(CC(NC(CC(C)SC)=O)C3)C2)=O)CC(F)(F)CC1C CCCCCCC(C)C(=O)NCC(C(C)C)NC(=O)CC(C)CC(=O)OC c1(C(=O)NCC(=C)CCNC(=O)C(CCC)OCC)ccc2ncccc2c1F Cc1cccnc1C(=O)NC1CCCN(C(=O)CC2(C)CCOC2)C1 C1(N2CCC(C(=O)Nc3c(C)cccn3)CC2)CCS(=O)(=O)C12CCC2 CCC(CC)CCC(=O)NCC(CC1CCCC1)C(=O)NC(C1CCN(C)C1)C C1(CNC(C2CC=C(C)CC2)=O)CCN(Cc2ccc3nonc3c2)CC1(F)F c1(SC)nc2ncnc(N3CCCC(NC(=O)C4=CCCOC4)C3C)c2s1 C1(CC(=O)NCCN(C(c2c(SC)cnn2C)=O)CC)CC2(C1)CC1(CCC1)C2 C(=O)(CC(C)(C(F)(F)F)N(C)C)N1CCC(NC(C(C(C)C)CN(C)C)=O)CC1 C1(CNC(c2ccc(CC)cc2)=O)CCN(C(=O)CCCc2ncco2)CC1C c1(CN2CCC(CNC(Cc3ccc(C)cc3)=O)C2)ccc(N(C)C)c(Br)c1 c1(OC)cccc(CN(C)C(C2(O)CCN(C(C)(C)C)C2)=O)c1OC c1(C(N2C(c3cn(C4(C)CC4)nn3)CCC2)=O)cccc(O)c1[N+](=O)[O-] C1(C2CCNCC2)(C(=O)NCCC(CCCC(C)C)C)CCOCC1 C12(C(=O)NC(C(C)SC)C)CCC(CC1NC(=O)CC1(C)CC1)C2 N1(C(c2ccn(C(C)C)n2)=O)CC2CC3CC2C1C3NC(C1CCOC1C)=O c1(OC)ccc2c(c1)CCCC2C(=O)N1C2CCC1C(CNC(=O)C(C)(C)C)C2 c1(C(N2CCCC(N(C(C3C(C=C)C3)=O)CC)C2)=O)cc(O)nc(O)c1 c1(N2CCCC(C3N(C(CC(C)(C)O)=O)CCCC3)C2)nc(C#N)ncc1Cl N1(C(C2(CC=C)CC2)=O)CCN(C2CCCN(C(=O)C(C)COCC)C2)C(=O)C1 N1(C(c2ccccc2N2CCCCCC2)=O)CCNCC1C(F)F C1(C(N2CCCC(F)CC2)=O)C2CC(F)C(C2)N1C(C1Cc2ccccc2N1)=O C1(C(N2CCC(N(C(c3c(C)cc(C)s3)=O)C)C2)=O)CCCCS1(=O)=O CC1CCN(C(=O)C(=Cc2cnn(C)c2)Cl)CCN1C(C1CCN(C)C(=O)C1)=O N1(C(c2c(CC)n(CC)nc2)=O)CCC(C)C(N(C(=O)CN2CC(F)(F)C2)C)C1 CCC(CC(=O)N(CC(C)NC(=O)CCNC(=O)CC(C)C)CC)C(C)C CCC(CC)C(C)C(=O)NCC1CC2CCC1N2C(=O)C(C)(C)CO c1(C(=O)NC(C)CCNC(=O)C(C)NC(c2ccco2)=O)ccn2c1CCC2 CCCCC(F)(F)C(=O)N1CCC(NC(c2ccnn2COC)=O)C(CC)C1 N1(C(CNC(=O)NC)=O)CCC2CC2(C(N2CCC(C(=O)OC)C2C)=O)CC1 Cc1cc(CNc2cccc(C(=O)NO)c2)c(C)n1-c1ccccc1.C=O C1(C(N(CCCCNC(c2csc(-c3ccncc3)n2)=O)C)=O)CNC(=O)N1C c1(C(N(CC(C)N(C(=O)C=CI)C)C)=O)ccsc1C(F)F CC(C)C(F)(F)CC(=O)NC1CCN(C(C2CC(O)(C(F)(F)F)C2)=O)CC1 C(=O)(C(C)(C)CC(C)C)NC(CNC(c1c(C)ccnc1C)=O)CC(C)C C1(C(=O)NCC(CCCC)NC(c2n[nH]c3c2CCC3)=O)CCC2(CC1)CC2 c1(CNC(C(C2CCC2)NC(CCOCCOC)=O)=O)ccc(Cl)cn1 C1(NC(CCCCC)=O)CC2CC1CN2C(c1cn(C)nc1C(F)(F)F)=O c1(C(=O)OCC)ccc2nc(C)n(C)c2c1.C12CC3CCC1(C3)NCc1cn2nn1 C1(C(N2C(C(N(CC(C)C)CC#C)=O)CCCC2)=O)CC2CCC(C1)O2 C1(Cn2cc(-c3c(C)n(C)nn3)nn2)CC2CC1N(C(=O)C(=O)C(C)C)C2 C#CCCC(C(=O)N1CCCC(C)(N(C)C)C1)NC(c1ccnn1C)=O O=C(CNC(=O)C(CC1COCCO1)C(F)(F)F)N=c1cc[nH]cc1 c1(C(=O)NC(C)C(C)(C)NC(=O)CC2CCCN2C)[nH]nc2ncccc12 c1(C(N(C)CC2CCCN(C(c3cc(C(N)=O)cs3)=O)C2)=O)ccc(N)cc1Cl C(C(CC(C)C)NC(C1CC=CCC1C)=O)NC(C(CC1CC1)OC)=O C1(C(N2CCC(N(C(=O)CSS(C)(=O)=O)CC)C2)=O)Cc2ccc(Cl)cc2C(=O)O1 c1(C(N2CC(COC)(CNC(=O)CC3(C)CC3(Cl)Cl)C2)=O)ncc(N)nc1C c1(CN2CCC(CC(N3CC4=CC(=O)SC4CC3)=O)C2)ccc2ccccc2n1 N1(C(C(C)SCCCC)=O)CCC(NC(=O)CC2CCC(O)C2)C1C C1(NC(C2=NOC(C)(C)C2)=O)CCOC2(CCN(C(=O)C=CC3CCC3)CC2)C1 c1(C(=O)NC2C(n3cc(C(C)NC)nn3)CCCC2)ccc2c(n1)NCC(=O)N2 CC1CCC(C(=O)NC2(CC(=O)NC3(c4ccon4)CC3)CCC2)C1 CC(C(C)(C)C)=CC(=O)NCC1OCCC1C(=O)NCCCCN1CCC1 C(=O)(C(F)C(C)(C)O)N(C(C)CN(C(=O)CSCc1cscn1)C)C C(=O)(C(O)C(C(C)C)OC)NCC(C(C)C)NC(C1(CC)CC1)=O C#Cc1cnc(C(=O)NCCCCC(N2CCSC3CCCC23)=O)c(C)c1 c1(OC)cc(CC(=O)NC2CC2NC(c2cc(N)ccn2)=O)ccc1Br n1(CC(C(=O)NCC(C)(C)NC(CC(COC)C)=O)(C)O)ccc(C)cc1=O c1(C(N2CC(CNC(C(C)(F)F)=O)OCCC2)=O)nc2cccnc2s1 C1(NC(c2c(C)con2)=O)CCN(C(c2ccc(-c3ccccn3)o2)=O)CC1O N1(C(COCCC)=O)CC2(CNC(C3CCC(O)CN3C)=O)CCC1CC2 N1(C(C(CC)CCOC)=O)CCC2CN(C(c3cccc4c[nH]nc34)=O)CC12 N1(C(CCCCCC)C(=O)NC(C)C)CCC(C2CC(O)C2)CC1 C12(C(=O)NC(CC(C)NC(CCc3cc(C)n(C)n3)=O)C)CCCCC1C2(F)F CN1CCC(C(=O)NC2C3COCC23)(NC(C2CCC2(F)F)=O)C1 Cc1noc(C(C)N(C)C(C2(C)CC(O)C2)=O)n1 c1(CC)cccc(C(=O)NC(C)CN(C)C(C2CC(=O)N(C(C)C)C2)=O)n1 CS(=O)(=O)CCCC(=O)NC1CCN(C(C2C3CC4C(C3=O)C24)=O)C12CCC2 c1(CC(=O)N(C(C)CNC(=O)CS(=O)CC)CC)ccc(C)cc1Cl C=CC1(C(=O)NC(CC(C)C)C(=O)OC)CCN(C(C2CN(C(C)C)C2)=O)C1 c1(C(N(C(C)CN(C(=O)CC(C)c2ccncc2)C)C)=O)cc(O)nn1C c1(C(N2CCOC(C3CCOCC3)C2)=O)cccc2ccsc12 N1(C(=O)Cc2cc[nH]n2)CCC2(CCCN2C(=O)CCCC2CCC2)C1 C(CO)(C(=O)Nn1ccnn1)NC(c1cc(C)nn1C)=O c1(C(=O)Nc2cc(OC)nn2-c2ccc(C)c(Cl)c2)cncc2ccccc12 C1(OCC(=O)NCC2CCCN(C(CC3C(C)C3(F)F)=O)C2)CCC(F)(F)CC1 N1(CCCC(=O)Nc2c[nH]c3ccccc23)CCC2(O)CCCCC2C1 C1(C(=O)NC(C2CCC2)C2CC2)CCN(C(c2cc(Br)ccc2F)=O)CC1O N1(C(C(C)n2cccc2)=O)CCC(NC(C2(CN(C)C)CC2)=O)C1 C=CC(C)(C)CC(=O)NC(C(C)NC(=O)C=Cc1cscn1)C(C)C C(=O)(C1=CC2CC(C1)CC2O)NCc1nc(CNC(C2(C)CSC2)=O)nc(O)c1 N1(C(C2(C(=O)OC)CC2C)=O)CC2(CCN(C(C3CC4CC4C3)=O)C2)C1 Cc1nn(-c2ccccc2)c(Cl)c1NC(C1CCCN1C(c1cccs1)=O)=O c1(C(=O)NC(C2N(C(CCNC(COC)=O)=O)CCC2)C)ccc2cc[nH]c2n1 Cc1c(C(=O)NC23CCN(C(=O)C(C)N4CCCC4)CC2C3)sc2ccccc12 C1(SC)CCN(CC2CC3COCC23)CC1 C1(O)(C(C(=O)NC(c2cnc[nH]2)C)NC(=O)CCN2CCCCC2)CCCCC1 C(=O)(CC1=NN(C)C(=O)C1)NCCNC(c1c(Br)ccc(C)c1)=O N1(C(CCC2C(C)(C)C2)=O)CC(F)CC1CNC(C1CCC(C)CC1)=O c1(C(=O)NCCN(C(c2cn(C3CCOC3)nc2C)=O)CC)cccc(O)c1 c1(C(=O)NCCN(C(C23CCC(C2)C3)=O)CC)cccc(CS(C)(=O)=O)c1 Cc1c(NC(c2ncn(C)n2)C)ncnc1NC(c1ncc(F)cc1F)C C1(NC(C2C(C)C2C)=O)CCN(C(c2ncccc2C2CC2)=O)CC1(C)C C=C(C)CCCC(=O)N1CC(C2CN(C(=O)C(C3CCOCC3)C)CCO2)C1 N1(C(CCC2CCCN(C)C2)=O)CCC2(NC(C3CC4CCCC34)=O)CCCC12 N(C1CCCCc2cc(Br)ccc21)C(=O)NCCNC(=O)OC Cc1cscc1C(N1CCC(CN=[N+]=[N-])C1)C(=O)NCc1cccs1 N1(C(C(Cn2cncn2)NC(COCC=C)=O)=O)CC(C2(C)CC2)C1 c1(CCC)nc(C(=O)NCC2(CNC(=O)COc3ccccc3)CCC2)co1 N1(C(Cc2cccc(C)c2C)=O)CCC(NC(C2(CCO)CC2)=O)C(CO)CC1 Cc1occc1CC(=O)NCCC1CCCN1C(C1(C2CCCO2)CCC1)=O C(C(CC(F)(F)F)NC(C1(C)CC(C(F)(F)F)C1)=O)NC(C(CC)SC)=O N1(C(c2cc(C)sn2)=O)CCC(C(=O)NCC2C=CCOC2)CC1 c1(C(N(CC)CC)=O)ccc(NC(C2CC2C(=O)NC(C)CO)=O)cc1Cl N1(C(C2CC(SC)C2)=O)C2CCC1CC(CCNC(=O)C=CC1CCOC1)C2 c1(C(C(=O)NC(CO)C(C)NC(c2ccc(CO)o2)=O)N(C)C)ccccc1Cl N#Cc1ccc(S(=O)(=O)NCC2CC(F)(F)CO2)cc1NCc1ncoc1C1CC1 C1(NC(CCSC)=O)CC(O)CN(C(=O)COc2c(F)cccc2F)C1 N1(C(=O)CC2(n3ccnc3)CC2)CC2C(C(=O)O)(C1)c1ccccc1S2(=O)=O C1(CNC(C(CCC)=CCC)=O)CCCC2CN(C(C3(C)CNC(=O)C3)=O)CC12 N1(C(C)C(N2CCCCC2)=O)CCC(NC(c2cc(C(F)(F)F)c[nH]2)=O)CC1 c1(C(N(C2CC(NC(=O)C(F)=C3CCCC3)C2)C)=O)cc(-c2ccns2)on1 C12(C(=O)OCC)CCC(C(=O)NCCCCCCCOC)(CC1)O2 C(=O)(CCCC1CCOCC1)N(CC(CNC(CCOCC)=O)O)C c1(C(=O)NCC2CCN(C(=O)C3=C(Cl)CCOC3)C2)ccc2nc(O)[nH]c2c1F N1(C(CC(=C)C)=O)CCC(C2CCN(C(c3cc(C(=O)OC)no3)=O)CC2)C1 C(C(=O)NCC1CC(NC(c2cc(-c3cccs3)[nH]n2)=O)C1)(C(C)(C)C)SC C1(OC)CC2CCC1CC2C(=O)NCC1(C)CCCN1C(c1ccsc1)=O C1(NC(C2(C(C)C)C(C(=O)OC)C2)=O)CCCN(C(=O)CC2CCOCC2)CC1 N1(C(COCCCC)=O)CCC2CN(C(c3ccc(C(C)C)c(F)c3)=O)CC12 c1(C(=O)NC(c2ccc(Cl)cc2F)C)cccc2c1CN(C(C1CN(C)C1)=O)CC2 c1(-c2cc(CNCCCNC(=O)OC)sc2)ccc(F)cc1 c1(C(=O)NC2CN(C(CC(CC)(F)F)=O)C(C)CC2)c(Cl)c2ccccc2n1C C1(CC)CN(C(c2cn(C)nc2C)=O)CCN1C(=O)C(O)Cc1cccc(Cl)c1 N1(C(C2(C(CC)=O)CC2)=O)CC(C(N2CCOC(C)C2CO)=O)C(C)(C)C1 c1(C(=O)Nc2cccc(-c3cc(C)nnc3O)c2)n[nH]c2c1CCC2C c1(OC(C(=O)N(CCNC(CCC)=O)CCOC)C)ccc(Cl)c(C)c1 c1(NC(=O)NCCN2CC(C)(O)C2)nnc2n1CCCCC2 C(C(N=c1[nH]ccn2nnnc12)C1CC1)NC(c1c(N(C)C)cccc1)=O N1(CCCOCC)CCCC(C)(NC(C2(C)C=CCCC2)=O)C1 C1(NC(Cc2ncc(C)s2)=O)CCCN(Cc2n[nH]c(C3CC3)c2C)C1 N1(C(CCC2CCC(=O)N2)=O)CCC(C2CN(C(C3(F)CCOCC3)=O)C2)CC1 CC1CC(N=c2ccn3c(Br)cnc3[nH]2)CCN1C(=O)CN1CCCCS1(=O)=O c1(C(=O)NC2CCN(C(C3(C)CCCCO3)=O)C2)cc(N)ccc1Cl Cc1ccc(NC(=O)CC2CN(Cc3ncc(Cl)s3)C2)c(C)c1C c1(C(=O)NC2CCC(CNC(c3cnsn3)=O)CC2)cn2ccccc2n1 c1(-c2nc(SCc3cn(C(C)C)nc3)on2)ccccc1C(F)(F)F CC(C)C(O)C(C)C(=O)NCCc1nc(C(=O)N(CC=C=O)C)co1 c1(C(=O)NC2C(C(=O)Nc3c(OC)nc(Cl)cc3)CCC2)cc(F)c(F)cc1C c1(CO)cc2cccc(NCC3CC4CCC3C4)c2s1 c1(C(=O)OC)c(C)cc(CN2CCCCC2C2CCCC2)cc1C N1(C(C(C2CC2)SC)=O)CCOC(C)(CNC(c2nnc(O)nc2O)=O)C1 C1(F)(C(N(C(C)CCO)C)=O)CCCN(C(C2CCOC(C)(C)C2)=O)C1 c1(C(=O)NC(C)(C)CCNC(C23CC(F)(C2)C3)=O)cc(C#N)c[nH]1 CC(C)CC(CN=c1cc(Cl)nc[nH]1)NC(=O)C(C)(O)C1CCC1 C1(NCC)CC(C(=O)N(C2CCC(NC(C3CCC3)=O)CC2)CC)CCO1 N1(C(C=C(C)C(F)F)=O)CC2CCC(NC(=O)C(c3cncn3C)O)C2C1 C1(C(N2CC(CC(C)NC(C3(N4CCCC4)CC3)=O)C2)=O)CCc2n[nH]cc2C1 C1(NC(c2c(-n3cc(-c4c(C)ocn4)nn3)cccc2)=O)CCCc2ccccc2C1 CCCC(C(=O)NC1C=CC(CO)C1)NC(c1cc(C(=O)OC)[nH]n1)=O c1(C(=O)NCCC(CC)(CC)NC(C2CC3(CCC3)C2)=O)nccc2n[nH]cc12 c1(C(N2CC3CC(NC(C4(C)C=CCC4)=O)C3C2)=O)cc(F)cc(F)c1O N1(C(CC=C)=O)CCC2(CCC(CNC(c3cc[nH]c3C3CCCC3)=O)O2)CC1 CC1=C(C(=O)O)CCN(C(C2CCCCN2C(=O)OC(C)(C)C)=O)C1 CCC(C)C(O)C(C)C(=O)N1CCN(C(=O)C(C)NC(C)=O)CC1C Cc1ccnn1C(C)C(=O)NCCCN(C(C1CC(CC(C)(C)C)C1)=O)C(C)C C1(C=C)(C(N(CCC=C)CC)=O)CCN(C(c2ccc(C)[nH]2)=O)C1 O=C1CCOC(C(=O)NCC=CCC(N2CCC(F)(C(N)=O)C2)=O)C1 C1(NC(c2c(CC)c[nH]n2)=O)CN(C(c2nccn3cnnc23)=O)CC12CCC2 C1(NC(CC2(CN(C)C)CCC2)=O)CCOCC1C(=O)NCCCn1cnnn1 N1(C(CN(C(C(C)C)=O)C)=O)CCC(C(=O)NC2CC(F)C2)C1C(C)C C1(O)(C(C)NC(=O)CS(N)(=O)=O)CCN(C(C23CC(F)C2C3)=O)CC1 C1(C(=O)NC2CCC(NC(c3c(SC)csc3)=O)C2)CCc2ccccc2O1 C1(C(=O)NC(c2nccs2)CC)CC2CNCC2C1 C#CC1CN(C(=O)C(CCOCC)NC(c2ccnnc2)=O)CCO1 S(=O)(=O)(c1ccc(C)cc1)N1C(C(=O)NCCNC(CCOC)=O)CCC1 c1(CC(C)NC(=O)C(N)=O)cccc(CNC(=O)Cc2coc(C(F)F)n2)c1 C(=O)(CC(C)CC(=O)N(C1CCCN(C(=O)C=Cc2ccsc2)C1)CCO)OC c1(C(C)=O)ccc(C(=O)NCCN(C)C(c2c[nH]nc2C2CCCCC2)=O)nc1 Cc1cnccc1C=CC(=O)NCCC(O)CNC(c1ccc(Br)cn1)=O C(=O)(C(CO)C(C)(C)C)NC1C=CC(CNC(c2cc(OC)ns2)=O)C1 C(=O)(CC(CC(C)C)NC(C1CC(=O)CS1)=O)N(C(CC)C)CCO C12(NC(c3cc(C)sn3)=O)CN(C(c3ccc(C(N)=O)o3)=O)CC1CS(=O)(=O)C2 c1(C(=O)OC)cc2oc(C(=O)NC(CNC(=O)C(C)C(C)O)CC(C)C)cc2[nH]1 C1(OC)CCCC(C(N2CC(C)(c3cn(CC4C5CCCC45)nn3)C2)=O)C1 Cc1ncc(C(=O)NC2CCCC2NC(c2c(Br)n[nH]c2C)=O)cc1C#N c1(C(N2CC(NC(C3ON=C(C(C)C)C3)=O)C2)=O)cnc(C(F)(F)F)c(Cl)c1 N1(C(c2n(CC)nc(C3CC3)c2)=O)CCC2CN(C(c3cnsc3)=O)CC2CC1 N1(C(C23CN(C(=O)CC4(O)CCCC4)C(CC2)CC3)=O)CCC2(CCCOC2)C1 C1(OC)CCCCC1CNC(c1n(CCCCCC)nnn1)c1ccccn1 N1(C(C(CCSC)O)=O)CCC(O)(C(C)NC(C2CCCS2)=O)CC1 c1(OC)ccc(-c2ccc(CN(CC(c3cccnc3)O)C)s2)cn1 CC(C(=O)NC1CCCC(NC(c2cc(F)ccc2O)=O)C1)C(F)(F)F C#CC1CN(C(=O)C(C(C)OC)N(C)C)CCN1C(c1ccc(Cl)cc1C)=O C1(NC(C2C(C)C2C)=O)CN(C(c2cc(N)nc(Cl)c2)=O)CC1S(C)(=O)=O CC(C(=O)NC(CC1CC1)C(=O)NCCC1=CCCCC1)C(F)(F)F C(=O)(CC(C)(C)CC(F)F)N(C(C)(C)C)C(N1CCN(C)CC1(C)C)=O CC1(C)CC(C(=O)NCC2CCCC2)CCN1C(C1CCC(C2CC2)C1)=O Cc1ccc(C(=O)NCC(C)(C)OCCNC(=O)CCc2nc(=N)[nH][nH]2)n1C CCC(C(=O)OC)C(=O)NCCCCCCNC(=O)CC1CCCOC1 C1(O)(CNCc2scc(C(N(CC(O)C3CC3)C)=O)c2)CCOCC1 Cc1c(C(=O)NCC(C)(CO)NC(c2cc(O)nn2C)=O)nnn1C(C)C C=CCCCCC(=O)NCCC1CCCN(C(=O)CC2CC(CC)C2)C1 C#Cc1cc(C(=O)NC2CCN(C(=O)C(F)F)C(C3CC3)C2)cc(Br)c1 C#CCCC(C(=O)NC1CCS(=O)(=O)C1)NC(c1cc(F)cnc1O)=O c1(C(=O)NC2CC3(CC(NC(C4CCC(OC)C4)=O)C3)C2)cc(C)c(C)cc1C N1(C(c2cc(C(F)F)on2)C(=O)NC2CCCC2)CCCC(C2OCCO2)C1 C(=O)(C1CCCc2cc(O)ccc21)NCC12OCCC(NC(C=CC)=O)(C1)C2 C1(CC)CN(C(C2(c3ccsc3)CC2)=O)CCC1NC(=O)C1=CCCCO1 c1(NC(CN2C(C)CCC2C)=O)ccc(Cl)c(Cl)c1.C12CCCN(C1)C2=O c1(C(=O)NCCN(c2cc(C(C)C)ncn2)CCC)ccc(C=NOC)cc1 c1(OC(C)C(=O)NCC2(F)CN(C(c3cc(C(F)F)no3)=O)C2)ccccc1Cl Cn1ccnc1CNC(c1n[nH]c(CO)n1)C1CCC1 c1(N2C3C(C(=O)Nc4c(C)c(Cl)ccc4)C(C3)C2)ncnc2c1CCC2 N1(C(c2cn3cc(C)ccc3n2)C(=O)NCCOC)CCCCC(S(C)(=O)=O)C1 N1(C(c2c(N)nccc2)=O)CCCC(NC(=O)CC(C2CC2)C2CC2)CC1 n1(C(C)C)ncc(Cl)c1C(=O)NCCC1CCCN(C(=O)CC2CC2(C)C)C1 C1(NC(c2c(C(C)C)ocn2)=O)CCN(C(c2cc(C#N)cn2C)=O)CC1O N1(C(CCCC(=O)N(C)C)=O)CCC2CCN(C(C3C4CCC3CC4)=O)CC2C1 c1(C(=O)NCCC(CCNC(C(C)(C)OC)=O)C)ccn2nccc2n1 C1(CC(=O)NCC2CC(NC(c3ccnn3CCF)=O)CC2O)CCCC1(F)F C(=O)(C1=CC2(CCOC2)C1)N1CCC(C(C)(C)NC(=O)C=C2CCCCC2)CC1 N1(C(C(c2ccc(Cl)s2)C)=O)CC=CC1CNC(=O)CCN1CCCC1=O c1(C(=O)NC2(CNC(=O)CCSCc3ccsc3)CC2)ccc2cnccc2n1 C(=O)(N=c1ccn(CCC)[nH]1)C1(CC=C)CCN(C(=O)C(C(C)C)NC=O)C1 C1(CNC(C2(SC)CC2)=O)(CNC(=O)CCCc2cnn[nH]2)CC12CCC2 n1(CC(=O)N(C)CC2C3CN(C(=O)CCC4(C)CC4)CC23)cnc2c1CCCC2 c1(C(=O)NC2C(C#N)CN(C(=O)Nc3ccccn3)C2)cc(F)c2cn[nH]c2c1 c1(C(=O)NC(C(C)NC(CC(C)C)=O)C)ccc(Cl)cc1 N1(CC(=O)NC(CSC)Cn2cc(C3(CO)CCC3)nn2)CCC(C)(O)C1 C(=O)(C(CCF)NC(=O)CCOCC(C)(C)C)NCC(C)SC CC1OC2(CO)CC1(C(=O)NCC1CCCN(C(c3ncc(F)cc3F)=O)C1)C2 C=C1CC2(C1)CN(C(=O)C=CCNC(c1coc(COC)n1)=O)C2 N1(C(CCC(CC)=O)=O)CC2CCN(C(C3C4CCCCCCC34)=O)C2C1 c1(C(=O)NCC(C2CCNC2)O)ccc(-c2nn[nH]n2)cc1Cl c1(OC)cc(C)c(C(N2CCC(NC(C3CC(OC)C3)=O)C2)=O)cn1 CCC(CC(F)F)C(=O)N(C1CCN(C(=O)C(C)=CC2CC2)CC1)CC CC1CNCCC1C(=O)N(C)Cc1ccccc1SC(F)(F)F c1(Cn2cc(C3(C)CN(C(=O)CCCC4CCCC(O)C4)C3)nn2)cccc(Br)c1 C(CCCCCNC(C1(C)CCNC1=O)=O)NC(C=CC)=O C1(C)(OC)CCCN(C(c2ccn(CCNC(c3cccc[n+]3[O-])=O)c2)=O)CC1 C1(N(C(=O)Cc2scnc2C)CC)CCCN(C(=O)CN2CCS(=O)CC2)C1 N1(C(CCCNC(C)=O)=O)CCCCC1C1CCCN(C(c2csnc2C)=O)C1 C1(C2(O)CCCN(Cc3cn4c(n3)C(=O)N(C)C4=O)C2)(C(=O)OC)CCC1 c1(C(N2C(C(=O)NCCC(CC)CO)C(C)CC2)=O)cc(C)c(O)nn1 C12(C(N3C(CNC(=O)C=Cc4cn[nH]c4)CCCC3)=O)CC3CC(CC(C3)O1)C2 C1(C(=O)NC2C(CCOC)C2)CN(C(=O)CC2CC(F)C2)CC1C(C)C c1(C(N2CC(CNC(CN(C(COC)=O)C)=O)C3C2C3)=O)nc(C)c(C)[nH]c1=O CCCC(C)(O)C(=O)NCC1CCC(CNC(c2ncc(N)nc2C)=O)CC1 N1(C(c2c(C)nns2)=O)CC2C(CNC(c3ncccn3)=O)C2C1 C1(C(=O)NCCN(C(C)C)C(C2CC(F)(F)C2)=O)CC2COCC(C1)C2(F)F C12(NC(c3ncc(OC)cn3)=O)CCCC1CN(C(c1nc(Cl)oc1C)=O)C2 N1(C(CC(=O)NCC)=O)CCN(C(=O)CN(C)S(N)(=O)=O)C(CC)C1 C(=O)(C1=NOC(C(N2CCCC2)=O)C1)NC1C(NC(CN2CC(=O)NCC2)=O)C1 Cc1nc(C2CC2)sc1CC(=O)NC1(C)CC(NC(C2CC(C)(C)C2)=O)C1 C12(NC(c3cnn(CC)c3Cl)=O)CCN(C(=O)C#CC3CC3)CC1C2 C1(CNC(C2(C#C)CCC2)=O)CN(C(=O)C(COC)CC)CCCO1 N1(C(C2CC(=C)C2)=O)CC(C)(C)CC1C(=O)NCCc1ncn(C)n1 c1(C(C)(C)C)ocnc1C(=O)NCCOCCNC(C1CCC(CN(C)C)O1)=O CC(CC#N)C(=O)N(C1(C(=O)NC2CCCSCC2)CC1)C C12(C(=O)NC)CCC(C(=O)N=c3[nH][nH]cc3C(=O)OC)(CC1)CC2 c1(C(=O)Nc2nc(C(N3CCC(C(=O)OCC)C3)=O)n(C)c2)ccc(Cl)c(O)c1 N1(C(c2[nH]cc(C#N)c2)=O)CC2CCOCC2(NC(=O)C2=CCCCCC2)C1 c1(C(N2CC(C(C)NC(=O)C(C)(F)F)C2)=O)cncc(F)n1 C1(C(C2CC2)NC(=O)NCC2CCCCS2(=O)=O)COc2cscc2O1 c1(COC)cnc(N2CCCC(NC(c3coc(Br)c3)=O)C2)nc1 C1(NC(=O)NC)CCN(C(c2nnnn2CCCF)CC2CCCOC2)CC1 CN1CCC(=CC(N2CCC(CNC(c3ccnc(Cl)c3)=O)C2)=O)CC1 c1(CC(=O)NCC2(NC(C3CCC4CC34)=O)CC2)cccc(Cl)c1F C1(CCC(=O)NCC2CCCCN2C(=O)CCc2cncs2)(OC)CCOCC1 n1(CC(=O)NCCCN(C(=O)COC(F)F)C2CC2)cncn1 CC1(NC(=O)Cn2cncn2)CCN(C(c2coc(O)n2)=O)CC1 C12(C(=O)NCCCCNC(CC3(CSC)CC3)=O)CC(C1)C(C)O2 C1(CNC(CCN(CCC)C)=O)CN(C(=O)C(F)(F)c2csc(=N)[nH]2)CCC1C C1(O)(C(C)NC(C2CCCC2c2nc[nH]n2)=O)CN(C(C2COC(=O)N2)=O)C1 C1(NC(C(CC)F)=O)CC2(CNS(=O)(=O)Cc3cccc(C(F)F)c3)COC1C2 C1(NC(CCN(C(CC)CC)C)=O)COCCC1CNC(=O)C(C(C)C)NC=O C(=O)(CCS(N)(=O)=O)NCC12N(C(c3c(=N)cc[nH]c3)=O)CC(C1)C2 c1(C(=O)NC2CN(C(C(C(C)(C)C)N(C)C)=O)CC23CC3)nc(Cl)c(=O)[nH]c1N Cc1cc(NC(N2CCC3(NCCN(S(C)(=O)=O)C)CCCC23)=O)ccc1C#N c1(OC)cc(C(N2CC(NC(c3c[nH]c(C)c3)=O)CC2(C)C)=O)ccc1C c1(-n2c(C(CSC)(C)NC(COc3ccccc3)C3CC3)nnn2)ccccc1Cl N1(C(C2CC(CC)(CC)C2)=O)CCCC1(C)CNC(=O)C(C)Oc1ccccn1 Cc1cnc(S(C)(=O)=O)nc1N1CC(NC(=O)CCc2ccsc2)CC(F)(F)C1 Cc1[nH]nc2ccc(C(=O)NC34CC(CNC(C5CC5C)=O)(C3)OC4C)cc12 Cc1sc(C2CCCN2C(=O)OC(C)(C)C)nc1Sc1csc(-c2cccs2)n1 C#Cc1ccc(C(=O)NC2(C(=O)NC3CCOCC3F)CCC2)nc1 O=C(N=c1[nH]n(CC(=O)Nc2cccnc2-n2cncn2)cc1Cl)N N1(C(CC2(C)CC2(F)Cl)=O)C2CCC1CN(C(=O)COC1CCCC1)C2 c1(C(N2CCC(N(C(CC)=O)C)C2)=O)ccc2c(c1)C(=O)CCC2 c1(CC(=O)NCc2c(C(N(C(CC)COC)C)=O)cco2)cccc(F)c1 C1(C(N2CCC(NC(CC(=O)NCC(F)(F)F)=O)C2)=O)CCC2(CCOCC2)O1 c1(NC(C)=O)ccc(N=c2ccn(CC(C)(F)F)[nH]2)cc1C(F)(F)F c1(C2(C(=O)NCC3C(NC(CCSCCC)=O)CC3)CC2)oncc1C C(=O)(C(C(C)(C)C)SC)NC1C(CNC(c2nc(CCC)oc2)=O)COC1 C#CCC(CC#C)C(=O)N1CCOCC1CNC(c1ccc(CC(N)=O)cc1)=O c1(C(=O)NC2CC2NC(C2CC2[N+](=O)[O-])=O)[nH]c2ccccc2c1Br N1(C(C(C)SCc2ccccc2)=O)CCC(C)C(NC(=O)CNC(N)=O)C1C C1(NC(c2cc(C(C)=O)[nH]n2)=O)COC2(CCN(S(=O)(=O)c3cccs3)CC2)C1 C1(C(=O)NCC2(CCC=C)CC2)(NC(=O)Cc2cc[nH]n2)CC(F)C1 c1(C(=O)NC2CN(C(CC(CC)OC)=O)C2)ccc2ccccc2n1 C(=O)(CCCOC)N(CCC(=O)NC(C)C(C)C)CC=C C(c1ccncc1C)=CC(=O)N(C(CN(C(C1N(C(=O)OC)CCC1)=O)C)C)C c1(CC(C)(C2CC2)NC(c2nnn(CC)c2C)=O)ncnc2c1c(Br)nn2C N1(S(C)(=O)=O)CCC(C(=O)NC(C2(O)CCCCC2)CNCC2C=CCC2)CC1 C1(NC(CCCCNC(C)=O)=O)C2CC3C1C3C2C(N1CCC(OC(C)=O)C1)=O CC1CCCN(C(=O)CC2(C)CN(C(c3nnc(O)nc3O)=O)C2)CC1 C12(CNC(C(CC(C)C)OC)=O)CN(C(=O)C=Cc3ccccc3)CC(F)(C1)C2 c1(C(C)NCCC(C)F)nccc(C(F)(F)F)n1 Cc1cccc2cc(C(=O)N(CC(C)(C)NC(=O)C=C3CCN(C)CC3)C)oc12 C(CC(C)C(=O)N(CCC(C(C)C)NC(c1csc(CO)n1)=O)C)=CCC C(=O)(NN=c1ccc2nccn2[nH]1)C12OC(C)C(CC1)C2 C(C)(CCCCO)C(N(C1(C(C)=O)CCC1)C1CCC1)=O.C12CC(=CC1)C2 N1(C(C=CC(C)NC(=O)C(C)(O)C2CCC2)=O)CC(=O)NC2(CC2)C1 C12(CNC(C(SC)SC)=O)CC(CCO1)N(C(C1C3CCC(C3)C1C)=O)C2 CCCCCCn1nnnc1C(c1csc(C(=O)OC)c1)NCC1CCC(=O)N1 c1(CC(=O)NCC2CN(C(C3CC(SC)C3)=O)CC23CC3)cnc2ncccn12 CS(=O)c1ccc(C(N2CCC(O)C(NC(=O)C(C)(C)C(N)=O)C2)=O)cc1 C1(N(C(=O)C(C)(C)NC(N)=O)C)CCCC(NC(=O)COC2CCCCCC2)C1 c1(C(N2CCC(NC(C3C(=C)C3)=O)C2C)=O)cnc2ccnn2c1C c1(CNC(COC(CC(C)NC(c2cccs2)=O)=O)=O)cc(F)ccc1O c1(CNC(C(n2cc(CNc3ccccc3)nn2)C)=O)ncc(Br)s1 C1(NC(=O)Cn2ccnn2)CN(C(=O)COCC2CCCO2)CC1n1cccn1 C(=O)(CCN=C(NCc1ncccc1OC)NCC(=C1CCCC1)F)NC CC1CC(C)(C)CCC1NCc1cc(S(=O)(=O)N(C)C)c[nH]1 CC1CCCN(C(C2CCCN2C)=O)C1CNC(=O)C=CCCc1ccccc1 C1(C(=O)NCCCN(C(C2(C)CN(C)C(=O)C2)=O)CCO)CC2(C1)CC1(CC1)C2 Cn1[nH]c(C(=O)NC2CCCCC2NC(C2CC2(C)C(F)(F)F)=O)nc1=O CN(OCC(F)(F)F)C(=O)C(c1cn(C)nn1)NC(C1(C)CCOCC1)=O c1(C(C)CNC(=O)C(C2CCCCC2)NC(C2OCCC2C)=O)ccc(CO)s1 N1(C(C2(C(=O)OC)CC2)=O)CC(NC(c2ccnc(N(C)C)c2)=O)C2(COC2)C1 c1(C(N2CC(OC)(CNC(=O)C#CC3(C)CC3)C2)=O)ccc2c(c1)CCC(=O)N2 c1(CC(=O)NCCN(C2CCCC2)C(=O)C=C2CC2)c[nH]nc1O c1(OC)ccc2[nH]nc(CN3CCSC(C(=O)Nc4cccnc4C)C3)c2c1 C1(NC(=O)C2=COCCC2)CC12CCN(C(c1cc(F)ccc1N)=O)CC2 C(=O)(C(C)(C)C(=O)NCCC1CCC(NC(=O)C(C)c2cncs2)C1)OC O=Cc1sc(CNC2CN(C(=O)CN3C(=O)CSC3=S)CC2C)c(Br)c1Br C(CCCCCC(=O)N1CCCC(N(c2ncc(F)c(SC)n2)CCO)C1)SC CCC(F)(F)C(=O)NCC(O)C(=O)NCCCC(C)O Cn1[nH]cnc1=NC(=O)c1nccc(NC(c2cc(C(F)F)ccn2)=O)n1 CC(C)CC(C)C(C(=O)Nc1ccc(F)cc1)N1CC(=O)NC(C)C1 c1(NC(C2CN(C(CC)C)C(=O)C2)=O)ccc(OC(F)(F)F)cc1C C1(CNC(Cc2c(CC)con2)=O)CC(C)CN(C(=O)CCC(=O)NC)C1 N1(C(C(CSC)C)=O)CC(C(=O)NCCCn2ccnn2)C(C)C1 C1(NS(CCC)(=O)=O)CC2CCC(C1)N2Cc1cncc(Br)c1C C1(NC(CSCCN(C)C)=O)CC2CC(C1)N(C(C1CC3CCC(C1)C3O)=O)C2 c1(CNC(C2(C#N)C(C)C2)=O)ccc2c(c1)CCN(C(=O)Cc1ccsc1)CC2 c1(N2CCCN(C)CC2)nc(=NCCCc2cncc(F)c2)[nH]c2c1CCCC2 C1(C(=O)NCCCCNC(C(c2ccccc2Br)OC)=O)C2CNC(=O)C12 N1(C(C(C(C)C)N(C)C)=O)C2CCC1CN(C(=O)C(=Cc1cn(C)nn1)F)CC2 c1(C(=O)OCC)ccc(C)c(C(=O)NC(c2nn(-c3ccccc3)nc2C)C)c1 CC(C)C(CC(=O)N1CC2(CC(NC(C3OCCN(C)C3=O)=O)C2)C1)C(C)C C#CCC(CC(=O)N=c1ccn(CC)[nH]1)NC(=O)CC1CCC(=O)N1C S(=O)(=O)(c1ccc(NCC(C)Cn2cccn2)c(Cl)c1)NC(CC)CO c1(C(=O)NCC(CN(C)C(c2csc(C(N)=O)n2)=O)(C)C)cc2[nH]ccc2s1 c1(C(=O)NC(CN(C(C2C(COC)(COC)C2)=O)C)(C)C)cc([N+](=O)[O-])oc1C C1(O)(CNC(C(CC)CC)=O)CCCN(C(C2(C#N)CC3CC3C2)=O)CC1 S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1CC(C)N(C)C(C)C1.c1(N)nc(Cl)cn2ccnc12 C=CC1CCCCN1C(C12CC1CCN2C(=O)C1=CCCCC1)=O Cc1ccccc1NC(C12CCCC1CC2)=O C1(Cc2ccc(N3CCOCC3)s2)CN(NCc2nc(C)sc2)CC1C Cn1cc(C(C(=O)NCCC(=O)NC(N)=O)NC(=O)Cc2ccc(Cl)o2)nn1 c1(C(=O)NC2(C)CCC(NCCOC3CN(C(C)=O)C3)C2)c(C)nc(O)nc1C C(=O)(C(C)(C)C1CCN(C(=O)CCc2cncnc2)C1)NC(c1cncs1)C N1(C(c2ccc(C(C)C)nn2)=O)CCC(CO)(CNC(C2C3CCCC23)=O)CC1 C(=O)(C#CC1CCCO1)NC(CCNC(C(CC)n1ccc(C2CC2)n1)=O)(C)C C(=O)(C1=COCCO1)N1CC(SC)C(NC(=O)C(C)c2ncco2)C1 c1(CC)cc(C)c(C(N2CC(C(C(=O)NC(c3ccc(C)cc3)C)OC)C2)=O)o1 C(=O)(C#CC1CCCO1)N1CC(NC(C2CCCCC23CC3)=O)C1 C1(F)(CNC(C2C(OC)CN(C(=O)CC3CC4C=CC3C4)C2)=O)C(C)(C)C1(C)C C1(C(=O)NCCCN(C(CC2(CSC)CC2)=O)C)CN(C2COC2)C1 C(=O)(C(CC(C)C)ONC(c1ccncc1F)=O)NCC(=O)NCC C1(C(N(CCCCC(=O)NCC2CCCC2O)C)=O)CCCC2(CC2)C1 C(CCC(=O)NC1CCC(CNC(=O)COC(C)C)C1)OCCOCC c1(SCCCC(=O)N2CC(CCNC(=O)CC3C=CCCC3)C2)ccc(F)cc1 N1(C(C(C)CC2CCC2)=O)CCc2c(CNC(C3CCCCS3)=O)cccc2C1 Cc1cc(C(N2CCC(C)(NC(C3CC(F)C(=O)N3)=O)CC2)=O)cc(F)c1C c1(NC(Cc2ncc(-c3c(C)cc(O)cc3)cn2)=O)c(Cl)ncc2ccccc12 c1(C(N(C)CC2(NC(C(CSC)O)=O)CC2)=O)cccc2c1NC(=O)CO2 C(=O)(CN=S(C)(C)=O)C(C(c1c(OC)cccc1)ONC(=O)C#CC1(C)CC1)=O c1(Nc2nccc(-c3cc(C)c(C(F)(F)F)cc3)c2)cccc2c1OCCC2 C1(OC)CC(C(=O)N(C)CCN(C)C(C)=O)N(C(c2cnc(Cl)n2C)=O)C1 c1(OC(C(=O)NCC2(CCNC(c3cc(C)oc3)=O)CC2)C)cccc(C#N)c1 Cc1cnn(C)c1CNC(=O)CN(C)C(c1csc(F)c1)=O N1(C(C(C)=CC2CC2)=O)C2CCC1CC(O)(CNC(=O)C(C)(O)C(C)C)C2 N1(C(c2cc(C)c(F)cn2)=O)CCCN(C(c2csc(Cl)c2Cl)=O)C(C)C1 C1(CC(=O)OC)CN(N(CC2CCCCO2)Cc2ccccc2)C1 N1(C(c2n(CCCCC)nc(C)c2)=O)CCCCC(N(C)C)C1 n1(CC)cc(Cl)c(C(N2CC=CC2CNC(c2ccnc(C(F)(F)F)n2)=O)=O)n1 c1(C(N(CCN(C(=O)C(n2cc(Br)cn2)C)CC)CC)=O)cccn1C c1(C(=O)NCC2OCCCN(S(CC(C)C)(=O)=O)C2)c[nH]c2c(F)cccc12 Cc1c(C(=O)NC2(CC(N3CCOC(C(=O)N(C)C)C3)=O)CCC2)cnn1C N1(C(Cc2c(C)non2)=O)CC2CS(=O)(=O)CC2(NC(=O)C=CC2CCCC2)C1 C(C)(CCCCNC(c1ncoc1C1CCC1)=O)NC(c1cc(CC)no1)=O S(=O)(=O)(c1cccnc1)N1C(C(=O)NCc2c(F)ccc(OC)c2)CCC1 C(CCCCn1cc(CCN(C)S(N)(=O)=O)nn1)NC(C(F)=C(C)C)=O N1(C(C2(C(N)=O)CC2)=O)CC(CO)(NC(C2CC(n3ccnn3)C2)=O)C1 N1(C(CNS(N(C)C)(=O)=O)=O)CC(OC)CC(NC(=O)Cc2c[nH]nc2O)C1 CC1COCC1N=c1nc2sccc2c(NCC(=O)N=S(C)(C)=O)[nH]1 CCS(=O)CC(=O)N1CC(NC(=O)C(=O)Cc2cccs2)CC1C N1(C(C2CN(C)C2)=O)CCCC2(NC(c3coc(Cl)n3)=O)CC2C1 N1(C(C2OCCN(CC)C2)=O)CCN(C(=O)C(CC)N(CC)CC)CC(C)C1 N1(C(c2cc(C(N)=O)[nH]n2)=O)CCc2c(CNC(C3CC34CC4)=O)cccc2C1 c1(C(N2CC(CC=C)(OCCC(=O)NCC)C2)=O)ccc2c(c1)C(C)C(C)O2 N1(C(C(C)OCCC=C)=O)CC2(CCCN(C(C3COCCC3(F)F)=O)C2)C1 Cc1cccc(C(N2C3CCC(C3)C2CNC(=O)Cc2c(C)n[nH]c2C)=O)c1C N1(C(c2ccn(C)n2)=O)CCC(CCNC(=O)CC2CC23CC3)CC1 CCCC(CC(C)C)C(=O)NC1(C(=O)NC2CCC3(CC3)C2)CC1(C)C N1(C(C(CCC)OC)=O)CCN(C(c2cnc(C3CC3)nc2O)=O)C(CCC)C1 C1(CC)CCCC1(C)C(=O)N(CC(C)(C)n1ccnc1)CC.C1C(C)=CC(=O)N1 c1(C(=O)NCc2ccoc2)ccc(-c2cscn2)cc1.C12(CC1)C(=O)NC2 c1(C(=O)NCC(CC=C)NC(=O)CCc2ncc(F)cn2)ccc(CC#N)cc1 CSC1=C(C(=O)NCCC2CCN(C(=O)CCCNC(N)=O)C(C)C2)CCCC1 c1(C(=O)NC2CCC2NC(C2CSC2)=O)cc2c(Cl)ccc(Cl)c2[nH]1 c1(OCCOC(c2ccc(-c3cc[nH]n3)cc2)=O)ccc(F)c(F)c1 C(CCC(=O)NO)NCC1CC(N)(C(F)F)C1 Cn1cnc2cc(CC(=O)NC(CNC(c3cc(O)cc(=O)o3)=O)CO)ccc12 Cc1c(C(=O)NC2CCC2NC(=O)CCCC(F)F)cccc1S(N)(=O)=O C1(CC(=O)OC2CCCC(SC)C2)CCc2ccccc2C1=O CCC(CC)(CO)C(=O)NCCC1CC(NC(C2CCC(=O)N2C2CC2)=O)C1 CCC(CCC(=O)N(C1CCCC1C#N)C)NC(=O)C(C)n1ccnn1 c1(CC)cc(C(N2CCS(=O)C(C)C2)C(=O)NC)ccc1OCC c1(C(=O)NCCC(C)N(C(CCc2cnc(C)o2)=O)C)ccc2c(c1)CCC=C2 N1(ONC(C=Cc2n(C)ncc2)=O)CC(C)(Cc2ccccc2)CC1(C)C c1(NC(C2CCN(CC3CC3)CC2)=O)ccc(Br)cc1O c1(C(=O)NC)ccccc1NC(C1CCCC1NCc1n[nH]cc1C)=O C(=O)(C(O)CNC(C)=O)NC1(C(NOCCCOC)=O)CCC1 N1(C(C2CN(C(C(C)SC(C)C)=O)CC2C)=O)CC(CO)CC(C)C1 C1(CC#C)(C(=O)NC2CCCC2CNC(=O)CSCC(F)(F)F)CC=CCC1 C1(CC(=O)N(CC(CC)OC)C)CN(C(=O)CN(CC(C)(C)C)C)CCO1 C12(CNC(C3(CC#C)CCC3)=O)CN(C(C3(C)CC=CCC3)=O)CC(F)(C1)C2 c1(C(N(C2CCC(CNC(CN(C3CCC3)C)=O)CC2)C)=O)cc(=N)[nH]c(Cl)n1 c1(CC(=O)N(CCNC(C(c2cccc(Cl)c2)C)=O)C2CC2)ccccc1Cl CC1CC(C)(C(=O)NC2CC(NC(c3cncc(OC(F)F)n3)=O)C2)CC(C)O1 Cc1nc(C(=O)C(=O)NC(C)(CNC(C2CC(N(C)C)C2)=O)CO)cs1 c1(CC(N2C(CN(CCCC=C)C)CCC2)=O)ccc([N+](=O)[O-])cc1 C=C(Cl)C(C)(C)C(=O)N1CCCC(C)(CNC(=O)CC(O)CCC)C1 C1(CC)CCN(C(=O)CC2(N(C(=O)Cc3ccc(F)c(F)c3)C)CC2)C(C)C1 C1(NC(C(=O)N(CC(c2ccccc2)O)C)=O)CC2CCC(C1)N2CC1CC1 Cc1ccc(C(N2CCC(NC(C3CC3c3cccnc3)=O)C(F)C2)=O)cc1Cl C1(C(N(C2CCN(C(c3cnn(CC)c3)=O)CC2)CCC)=O)CCCC(=O)O1 N1(C(C2CC3C=CC2C3)=O)C2CC1CN(C(C1(CO)CC1)=O)C2 CC(C)C(CCNC(=O)CC1CCCC1(F)F)NC(=O)C(C)OCC1CCCO1 CC1(C)COCCN1Cc1ccc(C(=O)NCc2cccnc2OCCO)cc1 c1(C(N2CCC(O)(CN(C(c3cc(OC)n[nH]3)=O)C)C2)=O)cc(N)c(F)cc1F C(=O)(CCC(F)(F)C(F)(F)F)N1CCC(C(C)NC(C2CCC(C)(C)CC2)=O)C1 C1(COC)(CO)CCCN(C(=O)COC(C2C3CN(C(C)=O)CC23)=O)C1.C(C)(C)C C=CC1(NC(=O)CC2CCN(C(=O)CCOCC3CCC3)CC2)CCOCC1 Cc1c[nH]c(C(=O)NCC(CC(C)C)NC(=O)C(C)Oc2cccnc2)c1C c1(OCC)cnc(NC(C(C)NC(c2n[nH]c(C)n2)=O)C(C)C)nc1 Cc1cc(CC(=O)NCCCC2CCCN2C(=O)C(=O)NC(C)C)ccc1CO Cc1ccc(CC(=O)NC(C2CCN(C(=O)C(C)NC(N)=O)C2)(C)C)c(F)c1 CC(C)C(CC(=O)N1CCOCC1CN(C)C(c1cnsn1)=O)C(C)C C1(C(=O)NC2CN(C(C3OCCC(=O)C3)=O)CC(F)C2)CCc2ncccc2C1 C1(C(N(CCC)CC)=O)(NC(=O)C(O)Cn2cncn2)CCCC1 N1(CC(N2C(C3(NC(=O)CN4CC=CC4)CC3)CCCC2)=O)CCCNS1(=O)=O Cc1ncc(C(=O)NC(C)(C)CNC(=O)CC2CCCC2O)c(Cl)c1Br C=CCC(CC=C)C(=O)NC1CN(C(=O)C(C2CC(C)(C)C2)OC)CC1C c1(C(N2CC(C)OC(C(=O)NCCN(C)C)C2)=O)cncc2ccc(F)cc12 C1(C(N2CC(CC(C)NC(=O)CCn3ccnn3)C2)=O)CCCCCCC1 N=c1[nH]c(C(=O)NCc2cn(CCNC(=O)CSc3ccccc3)nn2)cs1 C1(NC(c2ccc(C)s2)=O)CN(C(=O)Cc2ccc(Cl)cc2Cl)CC2CCCC12 C(=O)(C(C(C)(C)O)Nc1cccc(C(=O)O)c1)NCCC1C(C)(C)CCO1 C1(NC(c2ccc(CC)o2)=O)CCCN(C(c2cc(=O)n(C)cn2)=O)C1CC C=C(C)CC(C)C(=O)NCC1(C)CCC(NC(c2cn(CCCF)nn2)=O)CC1 CC(CCCCNC(=O)C(C1CCCO1)C1CC1)NC(=O)CC1CC(=O)NC1=O S(=O)(=O)(c1c[nH]ccc1=NCCC(=O)Nc1ccccc1)N(C(=O)CC1CC1)C c1(C(N2CCC23CCCSC3)C(=O)NC2(C)CC2)ccc2nccnc2c1 C(C(C(C)(C)C)NC(=O)CCCN1CCCCC1)NC(CCCOC)=O CC(=O)CCCC(=O)NCCC(C(C)(C)C)NC(=O)Cc1cn(C)nc1C(F)(F)F C(=O)(C(C)S(=O)(=O)C(C)C)NCCC(C)NC(C(CC(=C)C)NC(C)=O)=O Cc1cccc(N2CC(CN(C)Cc3cccc(CNC(C)C)c3)OC2=O)c1 C=CC1CN(C(=O)CCN(C(=O)COC2CCC2)C2CC2)CCO1 N1(C(C2(CCC)CCNC2=O)=O)C2CCC1CC(NC(c1cc[nH]c1)=O)C2 N1(C(C(C(C)C)F)=O)CC2(CCC(NC(c3cc(C(N)=O)co3)=O)CC2)C1 N1(C(C(CC)C(C)C)=O)CC2(CNC(c3ccco3)=O)CCC1CC2 CCC(Cc1ccccc1)CC(=O)NC(C)CCNC(=O)CC(O)CN(C)C C1(CCCCCC)CCCC1(c1nnnn1C(C)(C)CC)NCC=C(Cl)Cl C(=O)(C(C(C)(C)C(N)=O)NC(N)=O)N(C)CCNC(=O)CNC(=O)OC(C)(C)C CC(CC=Cc1ccccc1)C(=O)N(CCCCNC(c1ccsn1)=O)C CN1CCN(C(C2CCCN(Cc3cccc(I)c3)C2)=O)CC1c1ncc[nH]1 C1(CNC(=NCC)NCCCc2ccccc2Br)COC2(CCCC2)O1 CC1CCC(C(=O)NC2(c3ccccc3F)CC2)N1C(c1cnnc(O)c1)=O N1(C(CCN(C(CC)CC)C)=O)CCC(NC(=O)C=Cc2cncs2)C(O)C1 c1(C(N2CC3(CC(NC(c4cnc(SC)nc4)=O)C3)C2)=O)cc(C)c(Cl)c(C)c1 c1(C(N2CCCC(NC(=O)CC3CSCCS3)C2)=O)cc(F)cc([N+](=O)[O-])c1 C=C(C)C1OCCC1C(=O)NCC1CCC1NC(c1ccc(C(C)(C)C)nc1)=O CC1=NC(C(=O)NCC2(NC(=O)CC3CCC(C)C3)CCCC2)CS1 C(=O)(C(C(C)C)(C(C)C)SC)NC(CCCNC(C1CCC(OC)CC1)=O)C C1(NC(c2cc(C)ncc2C)=O)C2CCCN(C(C3CCCCS3)=O)C2C1(C)C C=CCC(C)(O)C(=O)N1CCC(CCC(N2CCOC(CC)C2)=O)C1 C(=O)(C1=CC2CCCC12)NCC1CN(C(c2n(CC)nnc2)=O)C(C)C1 C(=O)(CCCC(C)(C)NC(C1CCCC(=O)N1C)=O)N1C2C(C(=O)OC)C(C2)C1 S(=O)(=O)(c1ccccc1)C(=O)NCCCN(C(CC(C)F)=O)NCC1CCCC1 c1(C(C)C)ncc(C(c2nnnn2C2CCOC2)NCC(C)(C)OCCO)[nH]1 CS(=O)(=O)c1cccc(CC(=O)NC2(c3ccccc3)CCCN(C(C)(C)C)C2)c1 C(=O)(C#CC1CCCCC1)NCC(=O)NCC(N1C(CC)CCCC1)=O C1(NCc2c(C)nn(CCOC)c2C)CCC12CCCNC2 C(C(=O)NCC12CC(CNC(=O)CCC)(CO1)C2)(C(C)C)OCC c1(C(=O)NC(C2CN(C(=O)CC3CCOCC3(C)C)C2)C)ccn2cccc2c1 N1(Cc2ccc(OC)cc2F)CC(C2CCNC2)C1 C1(NC(C2C(CCC)C2)=O)CC2CCC(C1F)N2C(c1cnc(O)c(C)c1)=O c1(NC(C(=O)NCCN2CC=C(C)CC2)=O)cccc2nsnc12 C(CN=c1[nH]c(=NC2CCN(CCF)C2)c2cccc(F)c2[nH]1)C1CCN(C)C1 C1(CNC(Cc2cc(C)[nH]n2)=O)CN(C(c2csc(C)c2N)=O)CCC1(C)C c1(CC)cccc(C(=O)NCC2CCN(C(=O)CCSCC(C)C)CC2C)c1C Cc1nn(C)c(N)c1C(=O)NCc1n[nH]cc1C(=O)N(CC(O)CO)C c1(C(=O)NCC(C)NC(c2ccc(N3CCOCC3)cc2)=O)nc(=O)n(C)[nH]1 N1(C(c2c(C)ccc(C)n2)=O)CC2CCCC(C1)N2C(=O)CCCCN(C)C C#Cc1cnn(CC(=O)NCC2C3CN(C(C4CC4C(N)=O)=O)CC23)c1 N1(C(C2CC(C#N)C2)=O)CCN(C(C2CC3C=CC2O3)=O)C(C2CCCC2)C1 c1(C(=O)NC2C(CNC(CSCCC#N)=O)C2)coc2ccc(F)cc12 N1(C(c2cn(CC(C)O)c(=O)cc2)=O)CC(NC(=O)CC#N)C(C2CC2)C1 C1(O)(CNC(COC)=O)CCN(C(c2ccoc2Cl)=O)C1 N1(C(C2(CC)CC2(F)F)=O)CCC2CN(C(=O)C(C)(C)C3CCCO3)CC2CC1 C1(SCC(N2CCC(CC(C)CO)CC2)=O)CCc2ccccc2C1 C(c1ccccc1F)=CC(=O)N(CCCNC(C(=O)NCC)=O)C(C)C Cc1cc(C(=O)N(C(C)CN(C(=O)CCCc2cc[nH]n2)C)C)sc1C c1(C(=O)NC2CCN(C(C(CC)CC(C)C)=O)C2(C)C)ccc2cnccc2n1 O(NC(=O)C(C)C1CCN(C(=O)CC2CCSCC2)C1)C(C=C)C CC1=CCC(C(=O)N(C2CCC(NC(c3nnn(C)n3)=O)CC2)C)CC1 N1(CC(=O)NC(C2CC3(CCC3)C2)C)CCN(C(c2csc(CO)n2)=O)CC1 c1(C(=O)NC(CCCNC(c2cc(OCC)no2)=O)C)cc(F)cc(F)c1OC C1(C#N)(OC)CC(C(N2CCC2CNC(C2CC(=O)N(C)C2)=O)=O)C1 c1(C(=O)NC2(CNC(=O)CSCC(F)(F)F)CC2)nnc(O)nc1O c12cc(ccc1Cl)S2.c1(CS(C)(=O)=O)cn(CC2CCN2C(=O)CC2CCCO2)nn1 N1(C(c2cnc(CCCC)[nH]2)C(=O)NC2CCOC2)CCC(CCC(N)=O)CC1 N1(CC(=O)NC(c2ccccn2)=O)CCCCC1c1ccc(C(F)(F)F)cc1 N(C1CN(C(c2onc(C)c2C)=O)CCc2ccccc21)C(CC=C)=O c1(CN2CC(O)(CNC(=O)CC3CCOCC3)C2)c[nH]c2cccnc12 C(=O)(CS(=O)(=O)CC(F)(F)F)N1CCC(NC(c2n(CC)nnc2)=O)CC1C N1(C(C(C)(C)C2CCCC2)=O)CC2(CCCCN2C(c2cc(F)cnc2O)=O)C1 CC(C)CCC(O)C(=O)NC1CC2CC(NC(c3nonc3N)=O)C2C1 Cc1c(CN2CCN(C(C3CCCN3C(C)C)=O)CC2CO)oc2ccccc12 C(Cc1cnc[nH]1)(C(=O)NC(C)Cc1ccncc1)NC(CNC(CCC)=O)=O c1(SC)c(C(=O)N(C)CCOCCCN(C)C(C2CC3CCC3C2)=O)cnn1C CCCCCCC(CC)C(=O)N(C)CC1COCCN1C(c1ccc(C)cc1)=O C12(CCNC(C(C)N(C)C)=O)CCC(C1)N(C(c1ccc(Cl)nc1O)=O)C2 C1(C=C)(C(=O)NC(c2ccccc2)C#C)CCN(C(C2CC2(F)Cl)=O)CC1 c1(C(=O)NCC2(C)CCN(C(=O)Cn3cccn3)C2)ccnc2c(F)cccc12 c1(NCc2n(CC)nc(Br)c2)ccc(CN2CCCCC2)cc1C(F)(F)F CCCCCCC(C)C(=O)NC(C1CCCN1C(c1ccc(=NCC)[nH]c1)=O)C C1(NC(c2cn3c(n2)CCC3)C)CCCCN(C(=O)C(C)(C)c2ncco2)C1 N1(CCCNC(C2(CCC)CC2)=O)CCN(C(=O)CC(C)CC)CC1 C(=O)(C1=CC(C)CC1)NCc1ccc(CNC(C=CC)=O)cc1 c1(C(N(CCNC(C(CC)c2cccnc2)=O)C)=O)cc[nH]c(=N)c1[N+](=O)[O-] c1(CCC)cc(C(=O)NCc2csc(CNC(c3snnc3CC)=O)n2)n(C)n1 C1(C(N(C(C)C(=O)N(C2CCC2)CC2CC2)C2CC2)=O)CC12CCCCC2 c1(C(=O)NC2C3CC(NC(C(C)n4ccnn4)=O)CC32)cccc2oncc12 C1(C(=O)NCCN(C(C(=O)N(C)C)=O)C2CC2)CCN(c2nccs2)CC1 N1(CC(Cc2ccccc2)NC(c2ccc(Cl)cc2)C)CCCCCC1 CC1(CNC(C2CCCN(C(N)=O)C2)=O)CN(C2CCCNC2=O)CCO1 c1(C2(C(N3CCC(NC(C(CC)OCC)=O)CC3)=O)CC2)ccc(Cl)cc1Cl C1(C#N)(C(=O)NCC(C)C(F)(F)F)CCCOC1.c12cccc(c1)OC2 C1(NC(C2N(CC)CC2)=O)CC2(CCC(CNC(=O)CCNC(=O)CO)OC2)C1 C1(CNC(CCCC=C)=O)CC(C(C)C)CCN1C(c1cc(=O)cc(Cl)[nH]1)=O c1(CC)nn(C)cc1C(N1CCN(CC(=O)N(CC(O)CF)C)CC1)=O c1(OC)cc(Cc2ccc(-n3cc(-c4csc(C5CC5)n4)nn3)cc2)ccn1 C(=O)(CC(O)C(C)(C)C)NC(CCN(C(c1c(C)cncc1)=O)C)C(C)C C(=O)(C(C)CC(=O)OC)N(C1CCC(NC(CCCCC)=O)CC1)C C(=O)(C1CSc2ccccc21)N(C1CN(C(CCCC#CC)=O)CC12CC2)C N1(C(C=C)C(=O)OC)CCCC(C)(C(N2CCC2C=C)=O)C1 c1(OC)cc(F)ccc1C(N1CCCC(C)C1CNC(=O)Cc1ccsc1Cl)=O C1(CC)CN(C(C2CCC(C(C)C)N2C(c2nnc(S)n2C)=O)=O)CCO1 c1(SCCC(=O)NCCNC(Cc2c(C)occ2)=O)cc(F)ccc1F C1(CCOC)(C(=O)NCC(C2CCC2)NC(C2CN(C(C)C)C2)=O)CCCC1 CCCCC(C(=O)NCc1ccc(Cl)cn1)NC(c1cc(OC)n(C)n1)=O c1(CC)ncc(C(=O)NCC(C(C)C)NC(c2cn(C(F)(F)CO)nn2)=O)[nH]1 c1(C(N(CCCNC(=O)CC2SC(=N)NC2=O)CC)=O)cc(C)cc(OC)c1C c1(C(=O)NC(CC)CNC(C2(COC)CCOC2)=O)cc(OC)c(Br)s1 Cc1ccc(-c2ccc(C(N3CCCC3c3ccncc3C)=O)o2)cc1 C(CCC(C(=O)N(C)CC1CCCCCC1)NC(c1cc(C)no1)=O)OC N1(C(CSCCCC)=O)CCN(C(=O)C=CCCc2ccccc2)CC1C(F)F c1(CN2C(C(=O)Nc3c(C)nccn3)COCC2)cc(F)c(Cl)cc1F N1(C(CC2N(C(C(C)OC)=O)CCC2)=O)CC2CC(C1)c1ccccc12 N1(C(COCCOC)=O)CCCC(C2CN(C(=O)C(F)(F)c3ccccn3)C2)C1 C1(CNC(C(C)(C)n2cnnn2)=O)CC2(CO1)CN(C(C1(O)CCOC1)=O)C2 c1(N(C)CCOC2CC2)nc(N2CC3OCCOC3C2)nc2scnc12 C1(C(=O)NC2CCC(NC(c3cc(C(CC)CC)no3)=O)C2)CC2(CCCC2)C1 c1(C(N2CC(NC(CC(CC)SC)=O)C(C)(C)CC2)=O)cccc2[nH]cc(Cl)c12 c1(OC)cc(C)ccc1Cc1nccc(CC(=O)NC2CS(=O)(=O)CC2CO)n1 C=CCCCC(C(=O)N1CCCC(F)CC1)NC(=O)C(CC=C)NC(C)=O N1(C(CCCOC)=O)CCN(C(c2ccnn2C(F)F)=O)C2CCCCC2C1 C(CCC(O)CO)N(C(CN(C(CN(C(=O)OC)C)=O)C1CC1)=O)C C(c1ccccc1Br)=CC(N1CC(NC(C(COC)(C)OC)=O)C(C)C1)=O C1(CC)(NC(C(CCNC(C2CCNC(=O)C2)=O)OC)=O)CCCCC1 CC(CO)C(=O)NCC(O)CNC(=O)CC(c1cccs1)n1cccc1 C(=O)(CC(C(F)F)C(C)(C)C)N1CC(C)N(C(c2ccc(N)cc2F)=O)CCC1 N1(C(c2c(N)csn2)=O)CC(NC(c2ccc3ccoc3c2)=O)C2CCCCC12 N1(C(C2(NC(Cc3ccc(C)o3)=O)CC2(C)C)=O)CCCC2(CCCC2)C1 C1(CNC(C=C(C)C)=O)CC2(CO1)CN(C(=O)Cc1ccc(CO)cc1)C2 C1(NC(C(C(C)C)CO)=O)CN(C(c2ncccc2F)=O)CCC12CCOCC2 c1(C2N(C(=O)CCC3CCOC3)C2)ocnc1-c1cn(Cc2csc(Br)n2)nn1 N1(C(c2cnc(C)s2)=O)CC(NC(C23C=CC(CC2)C3)=O)C(O)C1 O=C1NCc2ccc(C(=O)NCCS(=O)(=O)Cc3cn(CC4CC4)nn3)cc2N1 c1(CC(=O)NCCNC(CN(C2CC2)CC)=O)ccc(Br)cc1C#N C12=NC(=NCCC3(OC)CN(C3)C1=O)NC=C2.c1(OC)ccc(CO)cc1 CCC(CC(=O)N1CCCC(C)(C(=O)NCCC(=O)NCC)C1)C(C)(C)C C(CN=C(NCc1nc(C)cs1)NCC(c1ncc(C)cc1C)C)SC c1(OC)c(C)nc[nH]c1=NCC1CCCCN(C(c2cnccc2C)=O)C1 N(C1COc2ccc(F)cc21)C(c1cncc(N)n1)=O c1(C(N2CC(C)C(NC(=O)COC3CCC3)CC2)=O)c[nH]c2cc(F)c(F)cc12 CC(C)(C(=O)NCC(O)CC(=O)N1CC2(CSC2)C1)C(F)(F)F C1(C2C(C(N(C3CN(C(C4CCN4C4CCCC4)=O)C3)C)=O)C2)CCCC1 C1(C(=O)NCCSC(C)C)CC(O)C(O)CC1CNC(C1CCN(C)C1=O)=O CC(O)(CC(=O)N1CCC(C2CCCCN2C(c2ccns2)=O)CC1)C(F)(F)F C1(NC(CC2C(C)(C)C2)=O)CN(C(=O)CSCC2CCCCO2)CC2(CC2)C1 c1(NS(C)(=O)=O)ccc(Br)cc1NC(N1CCCCC1CC1CC1)=O C1(C(N(C2CC(C(NOCC(=O)OC)=O)C2)C)=O)C2CCC(C2)C1C c1(C(N(CCCCCCNC(C2CC=CCC2)=O)C)=O)ccn2cccc2c1 S(=O)(=O)(c1cc(Br)ccc1Br)N1CCN(C(COC)=O)C2C1C2 C12(C(=O)NCC(CC)(CC)NC(c3cncc(N)c3C)=O)CCCCN1CCC2 c1(CC(=O)NC2CCCN(C(c3occc3Cl)=O)C2)cccc2nsnc12 Cc1snc2sc(C(N3CCC(NC4CCN(CC(C)C)C4)C3)=O)cc12 S(=O)(=O)(c1cnc(Cl)nc1)N1CC(CC)N(Cc2cc3ccccc3o2)CC1 c1(C2(C(=O)NCC3C(NC(CCCOC)=O)CC3)CC2)ccc(Cl)c([N+](=O)[O-])c1 O=C(C#CCNC(C1(CO)CCCC1)=O)NCCCC1CCCCC1 C1(OC)CC(CNC(=O)CSCC2CCCO2)N(C(=O)Cc2ccncc2C)C1 C(N=c1[nH]c(N2CCCC2)nc2cc(C(F)(F)F)ccc12)C1CCC(C)N1C N1(C(CCCC(=O)OCC)=O)CCCC2(NC(=O)CCc3ccccc3)CC2C1 CC(C)CC(C(=O)NCCC1(C)CC1(F)F)ONC(c1c(F)cncc1F)=O N1(C(c2c(OC)csc2)=O)CCc2sccc2C1CNC(C1(O)CC1)=O N1(C(CCC(=C)Br)=O)CCC2(CCN(C(=O)CCCC(C)CC)C2)C1 C(=O)(C(F)C(C)CNC(c1cn(CC)nc1C)=O)NC(CCC=C)C N1(C(c2ccc(CC)[nH]2)=O)CC(NC(c2cc(C)cnn2)=O)CC(C)(C)C1 N1(C(c2csc(C(F)(F)F)c2)=O)CCCC1CC(=O)NC12CC(OC(C)C)(C1)C2 N(C(=NCC(C)COc1ccccc1)N1CCC(C(=O)OCC)C1)CC(=C)C c1(OC)ccc(CC(=O)NC2CCC2CNC(=O)C=CC(=O)N(C)C)c(C)c1 C(N=c1nc(N2CCC(C)(F)C2)c2c([nH]1)CCCCC2)c1c(CC)nns1 CCCCCCC(C(=O)N1C2CCC1(CNC(=O)C1=CCOC1)CC2)NC(C)=O C1(CC=C)(NC(=O)C(C)NC=O)CN(C(=O)CNC2CCOC2)C1 CCCC(CNC(=O)COC(C)(C)C)C(=O)N1CC(CO)CC(C)C1 CCCCS(=O)(=O)CC(=O)NC1CCC(NC(=O)CCc2ccncn2)C1 N(C1CC2(CN(C(c3cc(C)c(O)c(N)c3)=O)C2)n2ccnc21)C(CCOC)=O c1(C(N2CC3C(NC(C4CCCCC(=O)N4)=O)C(C3)C2)=O)ccc2ccsc2c1 CC1c2ncc(C(=O)NCC3(O)CC3)n2CCN1C(c1ccc(Cl)nc1)=O CC1=C(C(=O)NCC2CCCN2C(c2nc(Cl)sc2Cl)=O)Cn2ncnc2N1C c1(N2CCC(c3onc(C)n3)C(C)C2)c(Br)c(C(=O)O)nc2ccccc12 C(c1ccc(OC)cc1)=C(C)C(N1CCCCC1C(C)(C)CNC(=O)CO)=O C1(NC(C2C(OCC)C2C)=O)C(C)CCN(C(=O)COc2ccsn2)C1C C1(N(C(c2c(C)cc(Br)o2)=O)C)CN(C(=O)C2=NNC(=O)C2)CCC1C N1(CC(N2C(CNC(CC(CC)O)=O)C=CC2)=O)C(=O)CC(C)(C)C1=O c1(C(N2CC(CCNC(=O)C=CC3CCC3)OCC2)=O)n[nH]c2cc(Cl)ccc12 C1(C(=O)NC2(CCNC(C3CCCC(O)C3)=O)CCC2)CC2(C1)CC1(CCC1)C2 Cc1cnc2n1CC(C(N1CC=C(CNC(=O)C(F)(F)C(F)(F)F)CC1)=O)CC2 C1(OC)CC(CNC(=O)CCC2CCCC(=O)N2)N(C(c2ncc(F)cn2)=O)C1 N1(C(c2csc3ccccc23)=O)CC2CCCC(C1)N2C(=O)CC1CCOCC1 c1(C(N(CCNC(C2C(C(=O)OC)CCC2)=O)CC)=O)cnn(C)c1C(F)(F)F CCCCC(CNC(C1(C)CCCO1)=O)NC(c1coc(OCC(F)(F)F)n1)=O N1(CC(=O)NC2(C(=O)NC(c3nc(CO)n[nH]3)C)CCC2)CCC(C(F)(F)F)CC1 C1(N(C)C(c2ccc(F)cc2)=O)CCCN(C(=O)C=CCN2CCCC2)CC1 N1(C(c2ccoc2Cl)=O)CCN(C(c2ccc(=O)n(C3CC3)c2)=O)CC2(CC2)C1 c1(NC)cnccc1C(N1CCCC(N(C(=O)CC2CCCC(=O)N2)C)C1)=O Cc1nc(C(=O)NC2CCCN(C(C3CN(C4CCOC4)C3)=O)C2)c(=O)[nH]c1C C1(NC(c2n(C)ccn2)=O)CN(C(=O)CCC2CNC(=O)N2)CC1n1ccnn1 C(=O)(C1Cc2ccccc21)NCC1CN(C(CCCN(C(=O)OC)C)=O)CC1O c1(C(N(CCC(OCC)OCC)CC)=O)cn(C)c(=O)nc1O c1(N2CCC(CCOC)C2)nc(=NCC(C)N2CCCCC2)[nH]c2c1CCCC2 N1(c2nc(C)c(C#N)cc2Cl)CCCC(C2CC2NC(=O)Cc2cc[nH]n2)C1 c1(C(C)C)cc(C(=O)NC(C2CCCC(c3ccccc3)O2)C2CC2)n(C)n1 O=C1CC(C(=O)NC2CN(C(=O)Cc3ccsc3)CC2C(F)(F)F)=NN1 N1(C(C(C)Cc2ccccc2)=O)CC(C(N2CCC23CCCC3)=O)CC(F)C1 C(CC(C)C)(C(=O)N1CCN(C(c2cnc(C)n2C(F)F)=O)CC1C)NC(C)=O N1(C(c2nc(C#C)sc2)=O)CCC(CO)C(NC(c2ccn(C3CC3)c2C)=O)C1 C1(O)(Cn2cc(CCOC)nn2)CCN(C(=O)C(F)CC2CC2)CC1 CCCC(C(=O)NCC(O)C1(Cl)CC1)NC(C1CCOC1C(C)C)=O c1(CC)noc(CC)c1CC(=O)NCCCCNC(=O)CCCCN1CCCC1 Cc1nc(C)c(C(=O)NC2CCC(NC(C3(C(F)(F)F)CCN(C)C3)=O)CC2)s1 c1(CC)ccc(C(=O)N(C(C)C(=O)NC2CC2(C)CC)C)[nH]1 c1(C(=O)NC2(C3N(C(CCCC)=O)CCCC3)CC2)cc(C2CC2)nc(O)c1 C(=O)(C1COc2ccccc21)N1CCC(N(C(=O)C2=CCC2)CC)C1 N(C1CCc2cccc3cccc1c23)C(c1cc(C)c(-c2cccc(Cl)c2)s1)=O c1(NC(CCOC)SC)nc(=NCC(C2CCCC2)SC)[nH]c2c(C)nn(C)c12 CCC(C)(COC)CNC(c1sc(Cl)cc1Br)c1nnnn1C1COC1 c1(-c2cn(CC(C)(C)CNC(C3C(CO)CCCC3)=O)nn2)cnccc1C#N Cc1nn(C)cc1-c1cn(NC(=O)NCC2(c3cccc(Cl)n3)CC2)nn1 N1(C(c2c(CC)n[nH]c2)=O)CCN(C(=O)CCc2cnn[nH]2)C(C)C1C N1(C(COc2ccc(C(=O)NC3CN(C(N)=O)C3)cn2)=O)CCC2CCC(C2)C1 c1(CC(N2C(C)(CNC(C(C)OC)=O)CCC2)=O)cccc(F)c1Cl C1(NC(C2OCCC(C)C2)=O)CC1C1CCN(C(C2CC3CC3C2)=O)CC1 C1(NC(c2c(CCC)occ2)=O)CCC(CNC(C2CC3CC2C3)=O)CC1 C(=O)(C(C)(F)C(C)(C)F)NCC(=CC(=O)N(C(C(=O)OCC)C)C)C c1(C(CNC(c2ccc(C)nc2)c2n(CC)nnn2)(C)C)ccccc1OC Cc1cc(C(=O)NC2CC(CCC(=O)NC(C)CN(C)C(C)C)C2)ncn1 C1(CC=C)(NC(=O)CCCOC(C)C)CCN(C(c2cscc2C(N)=O)=O)C1 O=C1CC2(CCN(C(C3CCN(C(=O)c4csc(Cl)c4)O3)=O)C2)CN1 C1(C(N(C)CC2CCCN2C(c2csnn2)=O)=O)CCn2c(O)nnc2C1 c1(-c2nnc(C3N(C(C)(C)C)CCOC3)o2)nc2cccnc2s1 N1(C(C(C)C2CC2)=O)CCC(O)(CCNC(=O)CCN2CCC(F)C2)CC1 n12cc(nn1)CCCC2.C1(C(C)NC(=O)C(=O)NCC(F)(F)F)CCCOC1 N1(C(c2ncn(CC)n2)=O)CC(NC(=O)CCc2cc(C)nc(C)c2)CC(C)C1 c1(C(=O)NC2CN(C(C(C)P(C)(C)=O)=O)CC23CC3)cc(S(N)(=O)=O)oc1Cl Cc1cc(Br)ccc1S(=O)(=O)N1CC2CC1CN2C(=O)CCC1CCC1 c1(C(C(=O)NC(c2cccnc2)C)N(C)CC2C3COCC23)ccc(F)c(Cl)c1 C1(CNC(C(C)OCC#C)=O)CC(CNC(c2csc(C(C)C)n2)=O)CO1 c1(CC(=O)N(C)CC2CCN(C(C(CSC)OC)=O)C2)cc(C(F)(F)F)nn1C C1(C(N(C)CN2CCOCC2)=O)COCCC1NC(=O)CSC1CCCC1 c1(C2CC(c3n(C)nnn3)(NC3(C)CC4(CCCC4)C3)C2)cc2cccc(F)c2s1 c1(CC(C)NCc2ccoc2C(c2nnnn2C)OC)ccccc1Cl N1(C(C=C(C)Cl)=O)CCN(C)CC1CNC(C1CCC2(CC1)CC2)=O C1(C(=O)NC(CC)CSC)(OC)CCN(C(c2coc(Cl)n2)=O)CC1 c1(N(C(COCC(C)C)=O)CCNC(=O)CCc2ccco2)ccccc1 C(=O)(C(CC#CC)NC(c1ccc(F)c(C)c1)=O)N1C(CCC#C)CCC1 CC1(C)CCCCC1(C)NC(C12CC1CCN2C(=O)CCn1cnc(=N)[nH]1)=O C1(NC(COCC(=C)C)=O)COC2(CCN(C(c3ccc(C(C)(C)C)[nH]3)=O)C2)C1 c1(-c2ccc(CN(CC(C)C)C)s2)cccc2c1nnn2C1CCCCC1 c1(OC)ccc(CC(=O)NC2(CN(C(=O)Cn3cc(C)cn3)C)CC2)c(Cl)c1 c1(C(N2CCC3(C(NC(COC4(C)CCC4)=O)C3)C2)=O)cc2ccsc2n1C c1(CC(N2CCN(C(c3n(CC)ncn3)=O)CC2C)=O)c(F)cccc1C#N CC(O)CC(=O)N(C(C)(C(=O)NCC1(C#N)CC1)C1CC1)C c1(OC)ccnc(C(N2CCC(F)C(NC(c3ccco3)=O)C2)=O)c1OC Cc1nnc2n1CCC2(C)C(=O)NC1COC2(C1)CN(C(=O)COCC1CC1)C2 c1(CC)onc(C(=O)NC(Cc2cc[nH]n2)C(=O)NC2CC2c2ccsc2)c1C C(=O)(CC(F)(F)C(C)C)N1CCCC(NC(CC2(CSC)CC2)=O)C1C c1(N(C)CC)nnc(-c2nc(C)n(C)n2)n1CC1CCN(C2CC2)C1 c1(CC)ncc(C(=O)N(C2CCC(NC(C3(Br)CC3)=O)CC2)C)c(C)n1 C(CCN=c1[nH]c(Cl)ncc1C)OCCNC(c1cc(C)oc1C(F)(F)F)=O c1(C(=O)NCC2CN(C(C3CCCCC3)=O)CCO2)cc2c(O)ncnc2cn1 N1(C(c2c(C)cn(C)n2)=O)CCN(C(c2cc(N(C)C)ccn2)=O)C2CCC12 C1(C#N)(OC)CC(C(N2CC(C)(NC(=O)Cn3cc(C4CC4)cn3)C2)=O)C1 c1(C(N2CCC(OC)(CNC(=O)CCS(C)=O)C2)=O)cncc(F)c1Cl N1(C(c2c(OC)ccs2)=O)CCCCC(NC(=O)CC2CC(OC)C2)C1 C1(CC(=O)OC)CC2(CCN(C(c3sc(=N)[nH]c3C)=O)CC2)CO1 c12ccc(cc1)C(=O)N(C)C2.C(=O)(CCC(C)C)NCC1CN(C(=O)NCC)C1 C#CCC(C(=O)NCC1(O)CCN(C(c2ccc(C(C)C)s2)=O)C1)C1CC1 c1(SC)ccc(C(C)NC(C2CSCCN2C(=O)CC2CCCCO2)=O)cc1 C(=O)(C#CC1(C)CCCO1)NCC1CCCCN(C(C(C)NC(N)=O)=O)CC1 C1(N(C(C2C(COC)C2)=O)C)CC2CCC(C1)N2C(c1ccccc1CC#N)=O c1(C(=O)NCC(C)CNC(=O)Cc2ccco2)cc(S(N)(=O)=O)ccn1 c1(CN2CC(F)(C(N3CCC(C(F)(F)F)C3)=O)C2)nc(Br)ccc1F n1(CC)c(C(=O)NCC2(O)CCN(C(=O)CCC(=O)OC)C2)cc2ccccc12 Cc1c(C(=O)NC2CN(C(C3CCN(C)C3=O)=O)C2)cccc1Br N1(C(CNc2c(C)cccc2)=O)CCC2(CC1)CC2C(N1CC2CC1CN2C)=O C=CC(CC)C(=O)NCCOC(C)(C)CNC(=O)C(CO)NC(N)=O C(=O)(C(O)CC(F)F)N1CCCC(NC(CN(S(C)(=O)=O)C)=O)C1 c1(OC)cc(OC)c(C(N2CC(NC(C3CC(C)(C)CO3)=O)C(O)C2)=O)cc1N CN1C(=O)CCC1C(=O)NC(C)(C)C(=O)NCCN1CCNC1=O C12(CNC(C34CCC3C4)=O)COC(CNC(C3COCCN3CC(F)F)=O)(C1)C2 C1(NC(CN(C)C)=O)CC2CC(NC(c3cc(SC(F)(F)F)c[nH]3)=O)C2C1 Cc1ncn(CCNC(=O)CCN(C(=O)C2=CCSC2)CC2CC2)c1C Cc1onc(C(=O)NCC(C)CN(C(=O)CC2OCCO2)C)c1Br C#Cc1cnn(CC(=O)NCC(c2ccc(F)cc2)NC(=O)C(COC)SC)c1 N1(C(CCC=CC)=O)C(C(=O)NCc2nn[nH]c2C2CC2)CC2CC12 N1(c2nc(C)cc(OC)n2)CC2CCC1C(NC(c1ccc(Cl)cc1)=O)C2 CC(CN=c1[nH]c(=N)[nH]c(=NCC2CC(O)C2)[nH]1)N(C)C(=O)OC(C)(C)C c1(C(=O)NC(C(C)C)(C)CNC(c2cc(Cl)ns2)=O)ccc2nncn2c1 C(=O)(CCCCN=[N+]=[N-])N(CCCCC(=O)NC(CCOC)CO)C c1(SC(C(=O)N(CCCCN(C(C2C(OC(C)=O)C2)=O)C)C)C)ccccc1 c1(C(N2CC3CN(Cc4c(C(=O)OCC)n[nH]c4)C3C2)=O)ccc(C#N)c(F)c1 C(C)(CCCCNC(C1(C)CCC(=O)N1)=O)NC(c1c(C)con1)=O C1(C(=O)NCC(C)NC(=O)COc2ccccc2Br)CCCCNC1=O c1(C(N(C(C)CNC(c2cn(C3CCC3O)nn2)=O)C)=O)nc(Cl)sc1Cl C1(C(C(C)C)NC(C=CC)=O)CCN(C(=O)CCSc2ccccc2Br)CC1 N1(C(C2C(C)(Br)C2)=O)CCCCC12CC(NC(c1ccc[n+]([O-])c1)=O)C2 C12(NC(c3c(C)cno3)=O)CCCC1N(C(=O)Cc1nn(C)cc1Cl)CCC2 O=C(C1=C(Cl)CCOC1)N1CCC1CNC(C12CCC(CC1)O2)=O c1(C(=O)NCC2CC(OC)CN2C(=O)C=C(C)Cl)cc2c(=O)cc[nH]c2s1 C12(C(=O)NCc3n(CC)ncc3)C(NC(C3CCC(=O)N3C)=O)C3CC1C2C3 C1(C(=O)NCC2CCCCC2O)CCN(C(=O)C=Cc2cccs2)CC1O C12(C(N3CC(O)(CNC(c4nccc(C)c4N)=O)C3)=O)CC3CC(C(=O)N1)C2C3 C1(N(C(=O)NC(C2CCOC2)C)C)CCN(c2ccccc2)CC1 NS(=O)(=O)c1cccc(C(N2CCCC2C2(O)CN(C(=O)C3=COCCO3)C2)=O)c1 C(C)(CC(C)N=c1ccnc(CO)[nH]1)NC(c1ccc(N(CCC)CC)cc1)=O c1(OC)c(F)cc(C(=O)NC2C3CC(O)C2N(C(C2CC(F)C2)=O)C3)cc1Cl N1(C(c2ccc(C)cc2Cl)=O)CCN(C(=O)CN2CC(C)C2)C2CCCCC12 c1(C(=O)NCC(C)N(C)C(c2ccc[nH]2)=O)ccc(C2CCCO2)[nH]1 c1(C(N2CC(NC(C3(CC)CC3)=O)C(C3CC3)C2)=O)cc2ccccc2cc1Cl N1(C(c2ccc(C(C)C)nc2)=O)CC2(CCCC2CCNC(=O)OC(C)(C)C)C1 CCCCC(C)(F)C(=O)N1CC(CN(c2ncnc(OC)c2OC)C)C1 c1(CNC(C(n2cc(-c3c(C)ccs3)nn2)C)=O)cc(Br)cc([N+](=O)[O-])c1Cl N1(C(C2CN(C)C(=O)N2)=O)CCCCC(N=c2ccc(C#N)n[nH]2)C1 C(=O)(CC(C)(C)CC(F)F)NC1CN(C(C2(C)CN(C)C(=O)C2)=O)CC1N=[N+]=[N-] c1(C(N2CCC(NC(CNC(CCCC)=O)=O)C2C)=O)c(Br)c(C)nn1C N1(CC=C)CCN(C(=O)CC2COCCN2C(C2CCCN2C=O)=O)CC1=O C1(CNC(c2ccn(C(C)C)n2)=O)CC(NC(=O)COC2CCCCC2)C(O)C1 C(C(=O)NC1CC2(C1)CC2C(=O)NCCc1c(C)noc1C)(C(C)C)OC CC1CC(NC(=O)Cn2nccn2)CN1C(C1COC(C)(C)C1)=O c1(C(=O)NCC2CCCN2C(=O)CSc2nncs2)ccn2nncc2c1 c1(NC(C(c2cccc(OC)c2)NC(C)C)=O)ccnc(F)c1I N1(C(C(CC)OC)=O)CC2CCN(C(=O)CCSC3CN(CC(F)(F)F)C3)CC12 CC1CC(N=c2[nH]c3c(c(=NCc4ncn(C)n4)[nH]2)CCCCC3)C1 N1(C(=O)Cc2ccsc2)CC2CCC(C1)N(C(=O)CCC(F)(F)C(F)F)C2 CC1CCCCC1(CNc1ncc(C(C)(C)O)cn1)NC(C1COC(C)(C)C1)=O C1(NC(N)=O)CCC2(CCC2)C1O.C12=CC=C(C=C1)C2 N1(C(C2N(Cc3ccn(CC)n3)CCC2O)=O)CCC2(CC1)CN(C)C2 c1(C(=O)NC2C(NC(CCc3nc(C)sc3)=O)CC2)cccc2cnccc12 c1(OC)ccc(CC(=O)O)cc1S(=O)(=O)N(Cc1ccccc1)CCl.C(=O)(C(N)=O)O c1(C(N2CC(C)(NC(Cn3ncc(CC)c3)=O)C2)=O)ccc(N)cc1Cl C1(C(=O)OCc2c(N(C)C)nccc2)CCC(=O)N(C(=O)CC2CCC2)C1 C1(CNC(C2CCN(C(C)=O)C2)=O)(CO)CCN(C(=O)Cn2cccn2)C1 C1(CC(=O)NCC(C2CC2)NC(=O)Cc2cccc(Cl)c2)CC2(CCC2)C1 N1(C(=O)CC2CCCCC2)C2CCC1CN(C(c1cc(-c3ccco3)no1)=O)C2 C#CCC(CC(=O)NC1(CCC=C)CCCCC1)NC(C1CCOC1)=O CC1(C(=O)NC2CN(C(=O)Cc3ccccc3Cl)CCC2CO)COC(=O)OC1 c1(CSCCC(=O)N(CCCCCNC(C2(C#N)CC2)=O)C)ccc(F)cc1 C(CC(C)CCNC(=O)C=Cc1csc(C)n1)NC(C(C)(C)SC)=O C1(NC(CC(CCC)O)=O)CN(C(c2ccc(C)s2)=O)C2(CCCCC2)C1 CCC1=C(C(=O)NCC2(n3cccn3)CCN(C(C3CC3=C)=O)CC2)SCCO1 N1(C(c2cnnc(O)c2)=O)CC2CCC1C1CN(c3ncncc3Cl)CC21 c1(NC(C2CN(C(C(=Cc3cn[nH]c3)C)=O)C2)=O)ccc(F)c(F)c1 Cc1ccc(C(F)(F)F)cc1C(N1CCC(C(C)NC(c2csnc2C)=O)C1)=O c1(NC(C(C)N(C(C(CCCC)C)=O)C2CCC2)=O)cnc2ncnn2c1 N1(C(CCC)=O)CCOC(CS(=O)(=O)Oc2ccccc2)C1 CC1(C)Nc2ccccc2C1NCc1ccccc1C(C)(F)F Cc1cn2c(C(=O)NCC(C)N(C(=O)CCC3CC3C)C)cnc2s1 C1(C)(CC)CC(C(=O)NC(C)CN(C)C(C2(C)CCCN2C)=O)CCO1 Cc1[nH]nc(O)c1CCNC(C12CC1CN(c1ncncc1OC(F)(F)F)C2)=O CS(=O)(=NC(=O)c1occc1)C1CC(O)C1.N1(C(=O)C2CC2)CCCC1 CCCC(CCCNC(c1cnc(S)[nH]1)=O)NC(c1nccn1CC)=O c1(C(=O)NCC(C2CCCC2)NC(C23CCC2C3)=O)cc2ccnc(Cl)c2[nH]1 c1(CC(=O)NC(C(=O)OCC)Cc2ccc(C#N)cc2)c[nH]c2cnccc12 C1(C(=O)NC(C(=O)NCC(C(=O)NC)C)CCN(C)C)CCCC12CCC2 C1(C(=O)NC(C2CCN(C(C3SC4C=CC3CC4)=O)CC2)C)CC2C(C1)C2(C)C O=C(C1OCCc2ccc(Br)cc21)N1CC(C2CC2)(CO)C1 c1(OC)cc(C(N)C(=O)NC2CC(c3ccccc3)C2)cc(OC)c1OC C(=O)(C(C(=O)NC(CC1CC1)CC(=O)N(C)Cc1cccc(O)n1)OC)OC C(=O)(C1=CCN(C(=O)C(O)(C2CC2)C2CC2)CC1)N1CCC(C)(OCC)CC1 c1(C(N2CC(C)(CCC(=O)NCC(C)O)C2)=O)ccc(C#N)cn1 C1(NC(=O)CC2COCCO2)COC2(C1)CN(C(c1ccc(O)c(F)c1)=O)C2 C(C)(C(C)S(C)(=O)=O)NCC(COC(COC)C)O c1(C(N(CCCC)C)=O)ccccc1C(=O)NC(c1ccccc1C)CO CCC(CN=C(NC1CCCC1)N1CCC2(C1)CC2(F)F)C(C)(F)F C1(NC(C2(C(=O)OCC)CCC2)=O)CS(=O)(=O)CC1NC(c1cc(C)[nH]n1)=O C1(CNC(C(=O)NCc2cccc(N3CCCCC3)n2)=O)CS(=O)(=O)CCO1 Cc1nnc(C(C)(C)NC(C2CC2C(C)NC(c2c[nH]nc2C(C)(C)C)=O)=O)s1 C1(CNC(C2(C(C)=O)CC2)=O)CN(C(=O)Cc2ncccc2C)CC1C N1(C(C(C)n2cccc2)=O)CCC2(CC(C(=O)NCC3CCCC34CC4)C2)C1 c1(C(=O)NC2(CNC(C3N(C)CCC3)=O)CCCC2)cnc(Br)c(N)c1 N#CC1(CO)CC12CCN(C(N1CCN(c3nc(Cl)c4cccnc4n3)CC1)=O)CC2 C=CC(O)C(=O)NC(CO)C(=O)NC1(CN(C)C)CCCC1 c1(OCC)cccc(CC(=O)NC2CN(C(=O)CSCCC#N)C3CC23)c1 C1(NC(c2cc(C(C)(C)C)no2)=O)CCCCC1CNC(C1(C)CC2CC2C1)=O N1(C(c2c(CC)nns2)=O)CCCCC1CCNC(C1SCCCS1)=O C1(C(N2CCC(C)(CNC(=O)C(F)=C3CCCC3)C2)=O)CCc2ncccc2C1 c1(C(=O)NC2CC3(CCN(C(CSCC(N)=O)=O)C3)C2)nncc2c1CCCC2 C(=O)(C(CNC(c1cnc(S)nc1)=O)C(C)(C)C)N(CCN(C)C)CC C(=O)(CC(C)NC(c1c[nH]c(=N)o1)=O)NCC(n1ccnn1)C CC1CCOC(C(N2CC(CC(C)NC(=O)C(C)(C)C3CCCO3)C2)=O)C1 C1(NC(c2cc(C)oc2C)=O)CC1C1CCN(C(=O)C(C2CC2)N(C)C)CC1 c1(C(=O)NC2CN(C(C3N(CC)C(=O)CC3)=O)C(C)C2)ccc2cccnc2c1 c1(C(N2CC(CC)N(C(c3cc(Cl)cs3)=O)CC2)=O)ccc2ncsc2c1 C(N=c1[nH]c(=NCCC2=CCCCCC2)[nH]c2c(F)cccc12)C1(CO)CCC1 N1(C(c2cccc(Cl)c2[N+](=O)[O-])=O)CCC2(CCN(C(C3CCCS3)=O)C2)C1 N1(C(CN(C)CC)=O)CCCC(C2CCN(C(C3(CF)CC4(CCC4)C3)=O)C2)C1 C1(C)(NC(=O)NCC(C(C)C)c2cccnc2)COc2ccccc21 C1(CC(=O)NC(C(C)Oc2cccc(C)c2)=O)CC2CCC1CC2(C)O c1(C(=O)NC2CC(N(C(=O)COc3ccon3)C)C2)cc[nH]c1-c1ccccc1 CP(C)(=O)C1CCCCC(c2nnnn2-c2ccccc2)(NCC2COC2)C1 N1(C(c2cncc(C#C)c2)C(=O)NC(C)C(=O)OC)CC(CO)CC(C)(C)C1 Cc1nc(Cl)cc(Cl)c1C(N1C2CC1CN(Cc1cnc[nH]1)C2)=O N1(C(c2ccc(OC)cn2)=O)CC2CCC(C1)N2C(C1(CC(F)F)CCC1)=O N1(C(C(CN(C)C)NC(C(C(C)O)N(C)C)=O)=O)CCC12CC(O)C2 c1(C(=O)NC(CC(=C)Cl)C(=O)N2CCC(C(F)F)C2)nccc2[nH]ccc12 Cc1cc(C(N2CCCC2CNC(C23CCOC(C)(C2)C3)=O)=O)c2c(c1)CCO2 c1(C(N2CC(CNC(C3CCCC3O)=O)OCCC2)=O)cc(F)c(O)c(F)c1 C1(C(N(CC(C)(C)CNC(=O)CCc2ccc(CO)o2)C)=O)CCCC(C#N)C1 c1(C(=O)NCCn2cc(CC(=O)OCC)nn2)ccc(-c2ccsc2)nc1 CCC(CCCC(=O)N1CCCCC1C(F)F)NC(C1CCN(CC)C1)=O c1(-c2cn(CCC(=O)NC3C(F)(F)C34CC4)nn2)cccc(Cl)c1Cl CCC(CC)CC(F)C(=O)NC(C1CC(NC(=O)C(C)CC2CCC2)C1)C CC(O)(CC(=O)NCC1(C(N)=O)CN(C(c2cnn(C3CCC3)c2)=O)C1)C1CC1 Nc1cc2c(cc1C(N1CCOC(CCNC(=O)Cc3cccs3)C1)=O)OCO2 Cc1cc(C(=O)NCC2CCC3(CCC3)C2NC(c2ccc[nH]2)=O)cn(C)c1=O CN1CC(C(=O)NCCCOC2CCN(C(c3ccc(N)cn3)=O)CC2)CC1=O C1(CC)CCN(C(C2CCC2CNC(=O)COC2CC2)=O)CC1 c1(C(=O)NC2CC(NC(C3(C)CCC3)=O)C2)cc(=O)cc[nH]1 c1(OC)c(C(=O)OC(C)C(=O)NO)cc(Cl)cc1C c1(C(=O)NCC(CC)NC(=O)CN2CC(C)(C)C2)cnc2c(c1)NC(=O)CN2 C1(CC)CN(C(=O)Cc2ccc(F)cc2)CCC1NC(c1cc(C)nc(C)n1)=O C1(NC(Cc2nc(C(C)(C)C)sc2)=O)CN(C(C2(CF)CC2(F)F)=O)CC12CC2 C(C)(C(CC(=O)N(C)CCN(C)CCO)NC(=O)CC1CCOC1C)OC Cc1cc2c(C(=O)NC3CN(C(c4cc(O)nc(Cl)c4)=O)CC3C)nccn2n1 Cc1ncc(Cl)c(C(=O)N(CCCCCNC(c2cc(F)ccc2O)=O)C)n1 C1(CCC(=O)NC(CNC(COCCCC)=O)CC)CCCCN1C c1(C(c2ccc(CC(=O)OCc3csnn3)s2)=O)ccc(Cl)cc1 c1(C(CC)CC)cccc(OC)c1.c1ccco1.N1(CC)CCN1 C1(CNC(=O)C=C2CCCCC2)CCCC1C(=O)NC1(CCO)CCC1 n1(CC(N2CC(NC(COCCOC)=O)C(C)CC2)=O)cnc2sccc2c1=O CCC(CNC(=O)C(c1cn(C)nn1)NC(C1CCCN1C1CC1)=O)(CC)CC N1(C(CNC(CC)=O)=O)CCOC(CC(N2CCC(F)(CF)C2)=O)C1 N1(C(C2CC(C)C2)=O)CC(Nc2cc(O)ncn2)CC2(CCC2)C1 c1(C(=O)NCC(=O)NC(CNC(c2c(CC)non2)=O)CO)cccc(OC)c1 C1(CCNC(=O)Cc2ccoc2)CN(C(C2CC3CC3C2)=O)CCS1(=O)=O c1(C(=O)NC2CN(C(c3c(C)coc3)=O)CC(C)C2)ccnc2c1ncn2C C12(NC(CNC(CC)=O)=O)CCCCC1N(C(c1c[nH]c(=N)o1)=O)CC2 CC1CCC(NC(c2csc(C(N)=O)n2)=O)CN1C(=O)COc1cccnc1 N1(C(CCCC2C(C)C2)=O)C(C(=O)NOC2CC3CCC2C3)CCC12CC2 Cc1nc(=NC(CNC(c2cccc(C#N)c2C)=O)CO)s[nH]1 N1(S(C(CC)C)(=O)=O)C2CCC1CC(NC(c1ccc(OC(F)F)cc1F)=O)C2 CC1CCN(C(=O)CCC2CCOCC2)C1C(=O)NC1CN(C)CC1C N1(C(C(C2CC(C)(C)C2)OC)=O)CC2C(CNC(C3CCC4(CCC4)C3)=O)C2C1 c1(OC)cncc(C(=O)NC2CCCC(NC(=O)CC3CSCCS3)C2)n1 N1(Cc2cc(C)no2)CCN(C(=O)NC(C(C)C)c2nc[nH]n2)CC1 CON=CC(=O)NCC1CCC(NC(=O)C(C)n2cccc2)C1 C1(NCCOCc2c(C)cncc2)CP(C)(=O)CC1O n1(CC(=O)NC2C(CNC(c3c(CC)con3)=O)CCC2)cc(C#N)cn1 CC(C)C(C)(O)C(=O)NC1CCCC1C(N1CCC(O)(CO)CC1)=O C1(COC)(CNC(=O)CCc2cn[nH]c2)CN(C(=O)COC2CC(F)(F)C2)C1 C(=O)(CC(F)(F)CS(C)(=O)=O)N1CC(C)C(CCNC(=O)CC23CCCC2C3)C1 Cc1ccc(C(N2CCCC(N(C(=O)CCC3CCOC3)C)CC2)=O)cc1C N1(C(c2ncc(OC)cc2F)=O)CCC2(CCCCN2C)C1 C1(OC)C(C(=O)O)C2CCC1(C)C2(C)C.C1(COC)(C)CN(C(=O)OC(C)(C)C)C1 N1(C(CN(C)CC)=O)CCCC(C)C1CNC(c1ccnc(F)c1N)=O CC1=CCN(C(=O)C=CC(C)NC(=O)OCc2ccccc2)CC1 C1(C(N2CCCC(O)(CCNC(C=CC(C)(C)C)=O)C2)=O)CN(CP(C)(C)=O)C1 c1(-c2ccncc2)cnccc1SCCC1CCCC1 C1(C(N2CCCC(c3cn(CC(C)(C)C)nn3)C2)=O)CC2CCC(C1)O2 c1(C(=O)NCC(C)NC(c2cc(SC)c(F)cc2)=O)ccc2c(=N)[nH]cnc2c1 c1(-n2c(C(O)C3CC3)nc(CC)n2)ccc(F)cc1OC c1(C(=O)NCC2(CNC(c3cc(C)n(C)c3)=O)CC2(F)F)ncc(N)cc1Cl C#Cc1cnn(C)c1C(=O)NCC1CC1CNC(C1(CC2CC2)CCC1)=O C12(NC(C3CCN(CC(C)C)C3)=O)COC(C1)C(NC(c1ccn(C)c1)=O)C2 c1(C(=O)NC)ccc(NC(C2CC23CN(Cc2c(Br)cnn2C)C3)=O)cc1 c1(C(N(C2CCN(C(c3csc(COC)n3)=O)C2)CC)=O)nc(C)oc1C c1(CC(=O)NC2(c3ccccc3)CN(c3ncccn3)C2)cnc(C(F)(F)F)cn1 CC(C)C(CCC(=O)NOCC1CC1)NC(c1ccc(O)cn1)=O N1(C(C2CCC(CC)CC2)=O)C2CCC1CN(C(C1C3CCC4C(C3)CC14)=O)C2 NS(=O)(=O)C1(C(=O)N(CCNC(c2ccc(O)nc2)=O)C2CC2)CC1 C1(NC(c2c(=N)[nH]cnc2)=O)C2CCC1N(C(c1cccc(C3(C)CC3)c1)=O)C2 C(=O)(C1CCCc2ccnn21)NCC1CN(C(C2CC(=C)C2)=O)CC12CC2 N1(CC(=O)N(CC(CNC(C2C(CCOC)C2)=O)C)C)CCc2sccc2C1 c1(C(C(=O)NCCN(C(=O)OC)C)NC(=O)C(O)C2CCC2)cccnc1 c1(C(N2CC(NC(CN(C)CC)=O)CC2(C)C)=O)cccc2c1OCC2 Cc1ccc(CC(=O)NCCN(CCCN(C)C)C(=O)CC2(C)CC2(F)F)cc1O C12CCN(CC1)C(=O)C1CCC1C(=O)N2CCC.N1(CC(=O)OC)CCC1C CC1CN(C(c2ccc([N+](=O)[O-])cc2)=O)CCCC1Nc1ncc(Cl)cn1 N1(C(CC2(OCC)CCC2)=O)CCC(C(=O)N(C)Cc2cn(C)nn2)C1C c1(C(c2nnnn2CCCOCC2CC2)NC(C)CCO)c(Br)ncn1C N#CC1CN(C(=O)C=Cc2ccc(O)cc2)CC1NC(=O)CCc1ccsc1 N1(CC(=O)NCC(C)(C2CC2)NC(C(C)N(CC(F)(F)F)C)=O)CCCCC1=O c1(C(N(C)CC2(CNC(=O)CSc3nc[nH]n3)CC2)=O)cnn2c1CCC2 c1(NC(C(C)C)CCN(C)C(c2cc(CF)on2)=O)nc(Cl)ncc1C1CC1 c1(C(=O)NC2(CC=C)CN(C(=O)C=Cc3cccnc3)C2)ccc(CSC)cn1 c1(C(=O)NCC2(O)CC(OCC)C2(C)C)oc2ccccc2c1Br C1(NC(c2ccc(C)cc2)=O)CC2CC1CN2C(=O)COc1cccc(F)c1 N1(C(C2C(C(C)C)C2)=O)CC(NC(=O)CNC(=O)COc2ccccc2)C(O)C1 CCCC1C(=O)N1.C1(CCOC(C)=O)CCN(C(=O)C(C)OCC)CC1 C1(NC(c2scc(C)c2Cl)=O)CCN(C(c2cc(Cl)cc(Cl)n2)=O)C(C)C1 N1(C(Cc2c(C)nsc2)=O)CCOC(C(C)NC(=O)COc2ccsc2Cl)C1 C1(C(N2CCCC(N(C(CC=CCC)=O)CC)CC2)=O)CN2CCCCC2CO1 N1(C(=O)COCC(F)F)CC2CCCC(C1)N2C(C1Cc2cccnc2C1)=O c1(OC)cc(-c2nc(C3CCOC3)nn2Cc2cnn(C)c2)cc(C(F)(F)F)n1 C12(CNC(C3CC(OCC)C3)=O)CC(NC(C3CCC(CC)C3)=O)(C1)C(C)O2 C1(NC(c2cc(C(C)(C)C)n[nH]2)=O)CCCC(NC(c2[nH]ncc2C#N)=O)C1 c1(CC(CC)C)nc(CC2CC2)n(-c2nc[nH]n2)n1 N1(C(C2(SC)CN(C(C(COCC)C)=O)C2)=O)CC(C)C12CCOCC2 N1(C(c2cc(C)n(C)n2)=O)CCN(C(c2ccc([N+](=O)[O-])n2C)=O)CC(CO)C1 C12(NC(COCC(=O)NC)=O)CCC(NC(C3COCCN3C)=O)(CC1)C2 C#Cc1cnc(C(=O)NCC(=O)NCC(N2CCC2C(C)O)=O)c(C)c1 NS(=O)(=O)c1ccc(C(=O)NCC(O)CCNC(=O)CC2CC=CC2)cc1 CCCC(CNC(=O)CN1CCCC1)C(=O)NCCCN1CCC(O)C1 c1(CC)[nH]c(C(=O)NC(CNC(C2CCCNC2=O)=O)CC(C)C)nc1Cl Cc1ncccc1C=CC(=O)NCCNC(C1(OC(C)C)CCCCC1)=O C1(NC(C=CSC)=O)CCC(C)(C)CC1CNC(c1cccc2c[nH]nc12)=O C1(C(N2CC3C(CNC(=O)Cn4cnnc4)(C3)C2)=O)CCCC(F)(F)C1 c1(C(=O)NCC(C)(C)NC(C2CN3CCN2CC3)=O)ccc(Cl)c(N)c1 N1(C(Cc2c(C)ocn2)=O)CC2(CNC(c3c(O)cccc3F)=O)CCC1CC2 CC1CC(C(=O)N)N(C(=O)CC2CCS(=O)(=O)C2)C1.C1(C=O)(CN(C)C)CC1 CC(C)CCC(O)C(=O)NCC(CC1CC1)C(=O)NC1(C2CCCO2)CC1 O=C(C1=NOC2(CCCN(Cc3ccc[n+]([O-])c3)C2)C1)N1CCN(C2CC2)CC1 c1(C(C(=O)NC2COC2)N(C(C)C2CC2)CC)cn(CC2CC2)nn1 Cc1cc(C)c2nc(N3CCC(C)C3CNC(c3ncccc3F)=O)sc2c1 C1(C)(CNC(C2(CC)CCC2)=O)CCC(NC(=O)Cc2ccccc2F)C1 Cc1cc(C(=O)N(C)CCN(C(=O)C(CO)NC(=O)C(F)(F)F)C(C)C)cn1C N1(C(C(CC2CCC2)OC)=O)CC(C(=O)NCC(C)F)C2(CC2)C1 N1(C(c2nn(CC)c(O)c2)=O)CCC(C2CN(C(C3CCC(C)C3)=O)C2)CC1 c1(OC)cc(C(N2CC(F)(CNC(=O)CNC(=O)CN(C)C)C2)=O)cc(F)n1 c1(OC)cc(CCCNC(=O)NCC(C(=O)O)C2CCOC2)ccc1Cl N1(C(C(C(C(C)C)O)C)=O)CC2CCN(C(c3nn(C)cc3[N+](=O)[O-])=O)CC2C1 c1(C(N2CCC(OC)(CO)C2)=O)cc2n(c1)CCNC2 c1(CC=C)ccc(C(=O)NC2CN(Cc3cnc[nH]3)CC2O)cc1 CC(C)(C(=O)NCCC1COCCN1C(C1OC2CCC1C2)=O)C(F)(F)F C(CC(=O)N1CC(C(=O)OC)C1)(C(C)CC)NC(c1n(CC#C)cnn1)=O c1(N2CCC(SC)C2)nc(=NCCC(C)c2cn[nH]c2)[nH]c2ccsc12 C1(OC)C(OC)CN(C(=O)C(=O)C(F)(F)F)C1CNC(c1cccc(=O)o1)=O C1(NC(CCC(=O)N(CCC)CC)=O)CN(C(=O)C2=CCOCC2)CCC1CO c12ccc(cc1)[nH]2.C1(C(=O)NC(CNS(C)(=O)=O)=O)CN(CCF)CC1F N1(C(C(F)OC)=O)CCCC2C1CCN2C(c1cc(-c2ccccc2)co1)=O C1(OC(c2cnc(S)[nH]2)=O)CN(C(=O)N(C2CCCOC2)C(C)(C)C)CC12CC2 c1(C(=O)NC2CC3(CCN(C(CC4CC(=O)C4)=O)C3)C2)ccc2nc(O)[nH]c2c1 CC(C)C(N=c1[nH]nc(C#N)s1)C(C)NC(=O)Cn1cc(C2CCC2)nn1 C1(c2n(CC(=C)C)nnn2)(NCc2cc(Br)no2)CC2CCCC12 CC(O)(Cn1ccccc1=O)C(=O)NC(CNC(c1csc(C(F)F)n1)=O)CO N1(C(C(CCC)NC(C)=O)=O)CCOC2(CCC(NC(c3cc[nH]c3)=O)CC2)C1 Cc1cc(C(=O)N(CC(C)CNC(c2cn(C)nc2C2CC2)=O)C)sc1Cl c1(N2CCN(C(C(C)OC)=O)CC2)ncnc(N2CCC(F)(CO)C2)c1C N1(C(C=Cc2c(C)ccs2)=O)CCC(CNC(C23CCCC2CCC3)=O)C1(C)C c1(CN2CCC(CC(=O)NCCOCCCC)C2)ccc(C#N)cc1 c1(C(=O)NC2CC(CC(=O)NC(c3ccccn3)CO)C2)cc(Cl)sc1Cl C(N=c1nc(N2CCC(C)(F)C2)c2ccc(C)cc2[nH]1)c1occ(C)c1 c1(OC)nc(Cl)ccc1C(=O)NC1CCCC(CN(C(=O)CNC=O)C)C1 c1(C(=O)NCCCC2(NC(=O)Cc3nc[nH]n3)CC2)csc2cncn12 c1(SCC(=O)NC2C(CNC(CCc3onc(C)n3)=O)C2)ccccc1Cl C(=O)(CS(=O)(=O)C(C)(C)C)N1CCC(C(C)NC(c2ccc(C(N)=O)cn2)=O)CC1 C1(OCC)CCCC1COC(=O)C(C#N)=CC1CC1 N1(C(C2N(CCC)CCC2)=O)CCC(F)(CNC(c2nocc2C(C)C)=O)C1 N1(C(c2ncn(-c3cn(C)nc3)c2)=O)CCN(C(c2cnns2)=O)C(CF)C1 N1(C(C2(Cc3cccnc3)CC2)=O)CCC2(CC1)OCCO2 C1(NC(CC2CCC(=O)N2)=O)CN(C(=O)CC2CC=CCC2)CC2(CC2)C1 N1(C(C=CC2(C)COC2)=O)CCC(F)(C(N2CCC(CC3CCC3)C2)=O)C1 C#Cc1cccc(C(=O)NC(CNC(=O)CC2(C(=O)OC)CC2)CC(F)(F)F)c1F C1(O)(C(N2CC(CCCCNC(C=CC=CC)=O)C2)=O)CC(CF)C1 c1(C(N(CC(CN(C(C(C)CCN(C)C)=O)C)O)C)=O)cccc2ccsc12 CC(C)CCCC(C)NC(c1ccncc1NCc1cnc(N(C)C)nc1)=O c1(C(N2CC(NC(C(CC)F)=O)C(c3ccccc3F)C2)=O)cc(Cl)ccc1F c1(CNC(c2n[nH]cc2Cl)=O)ccc2c(c1)CCN(C(C1C3CCC(=O)C13)=O)C2 c1(C(N(CC(C)NC(C(C(CC)(C)C)O)=O)C)=O)ccc2c(C)cc(Cl)nc2c1 C(CCC(=O)NCC1CCC1C(=O)NC1CC1c1ccn(C)c1)NC(C)=O C1(CNC(C2CCN(C)C2)=O)CC2CCC(C1)N2C(C1CC(n2cnnc2)C1)=O C(N=c1[nH]c(=NCC(C)F)c2cccc(F)c2[nH]1)c1ccc(C)c(N)c1 c1(C(N(C2CN(C(=O)CC3CSC3)CC2O)C)=O)cnn2ccncc12 Cc1cccc(CCNC(C2(NC(=O)C=CCCC(C)C)CC(F)(F)C2)=O)n1 C1(C(=O)OC)CCC(C(N2CCC(CNC(=O)CC3CCCCC3)C2)=O)CC1 C(=O)(C1=NOC2(CCC2)C1)N(C1CCC(NC(=O)C(C)(C)C#N)C1)C CCCC(C)(CC)C(=O)NCC1C2CC1N(C(=O)C=Cc1cn(C)cn1)C2 c12cc(c(Br)cc1OC)NC(=O)CC2.C(C(=O)NC1(COC)CC1)=CC Cc1cc(-c2noc(C(C3CCC(C)(C)CC3)(C)C)n2)ccc1I C(=O)(CCC[N+](=O)[O-])NC(CCCC)CNC(C1CCCN(C)C1)=O C1(C(=O)NCCC2CCC(NC(CSCC(=O)OC)=O)C2)CC1C1CCCCC1 N1(C(=O)C2=CCCCO2)CC2CN(C(=O)CCc3ccsc3)CC2C1 CC12CC1CCN2C(c1cc(CC2CCCCN2)on1)=O c1(N(C(CS(CC)(=O)=O)=O)C2CNCC2F)nc(C)nc2ccccc12 c1(CN2C(C(C)C)CN(C(c3cscn3)=O)CC2)c(F)c(F)c(F)c(F)c1F CC1CN(C(C2CC3(CC(NC(=O)C4=CCCCCC4)C3)C2)=O)c2ccccc21 c1(C(=O)NCC(CC=C)NC(c2conc2C(C)(C)C)=O)c(OC)cccc1C Cc1cc(C(N2CCN(C(=O)C(C)N3CC(C)C3)C(CO)C2)=O)c(Cl)cn1 C1(C(=O)NC(C(=O)NC(CN(CC)CC)C)C)C2CCC(C2)C1C FC1(F)C(CNC2C3CCC2CC3)CCC12CCOCC2 C(=O)(CCCS(C)(=O)=O)N(C1CN(C(c2ccc(O)c(F)c2)=O)CCC1O)C C(=O)(C(F)C(F)(F)F)NC(C1CCCN(C(=O)Cc2cscn2)C1)C N1(C(C(C=C)(C)O)=O)CCC2(CC(NC(C3(c4ccc(F)cc4)CC3)=O)C2)C1 C(CC(C(C)(C)C)NC(=O)C(N)=O)N(C(c1sc(C)c(O)n1)=O)C c1(-c2cn(CC)nn2)cncc(CN2C(=O)CCC2CNC(=O)CC2(CO)CC2)n1 CCC(C)(C#N)C(=O)N1CCC(CC(=O)Nc2cnn(C3CC3)c2)CC1 Cc1cccc(Cn2nc(C(C)C)nc2-c2ccc(COC)o2)n1 N1(C(c2cc(C)on2)=O)CC(C)OC2(CCN(C(c3cn(CCO)nn3)=O)C2)C1 C1(CNC(c2cncc(OCC)c2)=O)CN(C)CCN1C(c1ccc(Cl)[nH]1)=O CCCCCCC(=O)NC1CCC(CN(C)C(c2[nH]ccc2C)=O)CC1 N1(C(CCC(=C)C)=O)CC2(CNC(C3CC(O)(c4cccs4)C3)=O)CCC1CC2 N1(C(C(CC)N(C)C)=O)CCCC2(CCC2NC(C2CC(CCO)C2)=O)C1 c1(CC(=O)NCCC(C)NC(C2(C)CC2(Cl)Cl)=O)c[nH]c2cccnc12 CS(=O)(=O)c1cc(C(=O)NCCC2CCN(C(=O)C#CC3CCOC3)C2)co1 N(C(=NCCCCl)NC1CCC(N(C)C)C1)CCCSCc1cc(C)on1 c1(CN2CCC3(C(C(N4CC5COCC5C4)=O)C3)C2)cc(F)cc(F)c1Br N1(CC2(OCC)CCC2)C(=O)CCN(CC2CCCC(C)(C)O2)C1=O n1(CC(=O)N(CCCNC(=O)CC2CCCOC2)CC)nc(C)cc1C c1(C(=O)NCC2N(C(CC(C)n3cccc3)=O)CCC2)ccc(S(C)(=O)=O)[nH]1 c1(C(=O)NC(CC)CNC(=O)C(c2ccc(F)cc2)O)cc(C)n(C(C)C)c1C C1(C(=O)NC(C2CCN(C(C3CC34CCC4)=O)CC2)C)CC(C)(C)CN1C c1(NC(C(=O)N(C2CC2)Cc2ccc(C)cc2)=O)cc(Cl)c(Cl)cc1Br c1(CC)ccc(N)c(C(=O)NC2CCC2CNC(=O)C=CC2(C)CCOCC2)c1 N1(C(c2cc(COC)[nH]n2)=O)CCN(C)C(CNC(=O)CC2CCCO2)C1 C=CC1(NC(c2conc2CNC(=O)COC(C)CC)=O)CCCCC1 c1(C(=O)NCCCCN(C(CN(C)C(=O)C2CC2)=O)C)ccc(F)c2occc12 Cc1cc(Br)c(I)cc1NC(C1CC1c1ccccc1C)=O C1(NC(c2n(C)nc(O)c2)=O)CN(c2cnc(C#N)cn2)CC2(CCC2)C1 C(=O)(CCCCCOC)N1CCC(N(CC#C)C(C2CCC2COC)=O)CC1 C1(CNC(c2cccnn2)=O)CCCCC1C(=O)NCC.C(C(F)(F)F)OCCO CN=c1[nH]cc(C(N2CC(C(C(N3CCOC(C4CCC4)C3)=O)OC)C2)=O)o1 N1(C(c2nc(OCC)oc2)=O)CC(C)CN(C(=O)CC#N)C(C)C1 CC1CN(C(c2ccc3nonc3c2)=O)CCCN1C(=O)CC1CCCOCC1 c1(C(=O)NC2CCN(C(C(CC=C)CC=C)=O)C2)cc2ccc(COC)cc2[nH]1 [N-]=[N+]=NC1(C(=O)NCc2ccc(O)cc2F)CCN(C(=O)CCCC2CC2)C1 c1(C(CNC(=O)C=CCN2CCOCC2)NC(C2C(C)C2)=O)cccc(Cl)c1 C1(C(N(C2CSC2)C)=O)C2CC3C(C2NC(=O)C2=C(Cl)CC2)C13 C=CCC(C(=O)N(C(C)CN(C(=O)CCCc1ccc(O)c(F)c1)C)C)C(C)C c1(OCCOC)ccccc1NC(=O)NCC(O)C(F)(F)F C1(NC(C(CC=C)NC(=O)CC2OCCO2)=O)CCCOC12CCC2 N(C(=NCCc1ccnc(C(C)C)n1)NC(C)C)CC1(C(=O)OC)COC1 c1(C(C(F)(F)F)NC(C2N(Cc3cnc(C)s3)CC=C2)=O)cccc(F)c1 c1(OC)cc(C)ccc1C(N1CCCC1CNC(=O)C(c1ccc(F)cc1)F)=O C(=O)(CC1CCOc2ccccc21)NCC(C)NC(c1cc(=N)[nH]c(Cl)n1)=O c1(C(N2C(CNC(c3ccoc3Cl)=O)C=CC2)=O)ccc2nc[nH]c2c1 CCCCC(F)C(=O)NCC1CN(C(c2c[nH]nc2OC)=O)CC12CC2 C1(NC(c2cc(CN(C)C)no2)=O)CCCC(NC(c2cn(CCF)nn2)=O)C1 N1(C(C2OCCC(NC(C=CC(C)(C)C)=O)C2)=O)CCc2ncsc2C1 Cc1ccc2nonc2c1C(=O)NCc1ccccc1CNC(=O)CCCCCO CC1CN(C(c2cnsn2)=O)CCC1C(=O)Nc1cncnc1O N1(C(c2cc(C)sc2)=O)CC(NC(=O)C(C)Cn2cccn2)CC(F)C1 c1(C(=O)NCCOC2CCN(C(CC3CC(SC)C3)=O)C2)cc2c(s1)CCC2 C1C(C)(C)CC(=O)N1.Cc1cc(CCCCCN2CCOCC2)n[nH]1 C1(C(=O)NC2CN(C(CC)=O)C2)CC=CC(NC(C2CCN2C)=O)C1 c1(OC)c(C(N2CCN(C3CC3)C(C)C2)C(=O)NC2CCOC2)cccc1O c1(C(=O)NCC(C)CN(C(=O)CC2CCCCC2O)C)cn2cc[nH]c(=O)c2n1 c1(OC)cncnc1Nc1cccc(NC(C)=O)c1.c12nc(C)c(s1)c(=O)[nH]2 CC(C)C(CCN(C(=O)C(C)(C)C1CCCO1)C)NC(=O)C(O)CC1CCCC1 c1(C(N2CC(NC(C(CC=CC)C)=O)C(O)C2)=O)ccc(S(=O)(=O)CC)cc1 CC(C)CC(CNC(c1ccc(C(N)=O)o1)=O)C(=O)N(C1CCN(C2CC2)C1)C C(CC(=O)NC1CN(C(N)=O)C1)(C1CC1)NC(C1CC(OCC)C1)=O C1(C(=O)NCCN(C(COCC=C)=O)CCOC)CCc2ccccc2C1 C1(N(C(CC2CCN(C)C2)=O)C)CCCN(C(=O)CCn2ccccc2=O)C1 N1(C(=O)C=C(Cl)Cl)CC2CC(NC(C3(C4CCCO4)CCOCC3)=O)C1C2 c1(C(=O)OCC)nc(N2CCCC2CC(=O)NCc2conc2CC)sc1Cl CC1CC(C(=O)NCC2CC3(C2)CN(C(=O)CN(C)C)C3)CCS1(=O)=O c1(C(N(CCn2cc(-c3ccon3)nn2)CC)=O)cc2c(OC)cccc2s1 c1(CCC)n[nH]c2ccc(C(=O)NCC(F)CNC(C3CCOC(=O)N3)=O)cc12 N1(CC(=O)N(CCC#N)C)CC23CCCCC2(COC3)C1 c1(CC(=O)OCC)noc(C(C)NC2CCOC2)n1 N(C(=NCCN1CCCC1)N(C)Cc1cc(F)ccc1C)CCC(C)=O C(=O)(C(CC)CCCCC)N(CC(=O)NC1CN(C)C(C)(C)C1)CC#C c1(OCC(=O)NC2CCCCC2CNC(c2nsnc2O)=O)ccc(Cl)nc1 N#Cc1nccnc1N1CCC(CNC(c2ccc(-n3cncn3)nc2)=O)CC1 C(=O)(C1=CCC2CCC1N2C(c1cnn(C2CC2)c1)=O)N(C(C)CO)C C(=O)(C1COc2ccc(F)cc21)N1CCN(C(=O)CCc2cc[nH]n2)CC1CO CCCC(CC)CCC(=O)NC1CCCC(NC(=O)C2=C(Cl)CCOC2)C1 c1(CC)oc(C(N2CCCC2CNC(C2C(C)(C)C2(F)F)=O)=O)cc1C S(=O)(=O)(c1ccccc1C(F)(F)F)N1CCC(C(=O)Nc2cnn(CCO)c2)C1 C1(NC(C2(C=C)CCC2)=O)CC(OC)CN(C(c2nccn2CC)=O)C1 c1(C(CCO)NC(c2cscc2I)=O)ccccc1Br N1(C(C(C)(C)NS(C)(=O)=O)=O)CCC(C2CCN(C(C3(O)CCSC3)=O)C2)CC1 C(C(C)C(F)C(=O)NC1(c2cnc[nH]2)CC1)NC(C(C)OCC)=O c1(COCC(N2CCC(OCC(F)F)C2)=O)cccc(Cl)c1 c1(OCCOC)ccc(C(N2CC(C(C)NC(C3CCCC3C)=O)C2)=O)cc1 c1(SC)cc(C(N2CCCC2CN(C(=O)CC(C)(F)F)C2CC2)=O)ccn1 c1(OCCN(C)C)cccc(C(N2CCCC2(C)CNC(c2cnsn2)=O)=O)c1 C1(C(N2CCCC(OCCC)C2)=O)CC2CCC(C1)N2C(c1cc[n+]([O-])cc1)=O CON1CCC(CC(=O)NC(C)CCCNC(=O)CC23CC(C2)C3)CC1 n1(CCCC(=O)NC2CCC(CNC(CC3(C)CC3(F)Cl)=O)C2)ccccc1=O n1(CC(=O)N(C2CCN(C(=O)COC3CC3)C2)CC)ccc(Br)n1 c1(CC(N2CC(C)(CNC(CSCCOC)=O)C(C)C2)=O)cc(F)c(C)cc1F N1(C(c2c(C)occ2C(F)(F)F)=O)CC(NC(C2CC(CF)C2)=O)CC(O)C1 C1(C(=O)NCCc2c(C)n[nH]c2C)CN(C(c2cccc(=O)o2)=O)CC1(F)F C1(NC(CCC)=O)CC(F)(CNC(=O)COCC(N2CCCC2)C)C1 C12(C(N3CC(C(=O)OC)C3)=O)CCN(C(=O)C3=CCCC3)CC1C2 c1(C(=O)NC2CC(CNC(CCCC#N)=O)C2)ccc(S(=O)(=O)NC2CC2)o1 c1(N2CCC(c3n(C)cnc3)CC2)nccc(=NC(CCO)c2cccc(F)c2)[nH]1 c1(COC)cc(C(=O)NC2(CO)CN(C(=O)C(C3CCCOC3)OC)C2)cs1 C(=O)(C1=CCN(C(C2(C)CC2(C)C)=O)CC1)NC(C)Cc1cnccn1 C1(C(C)C)CCC(C(=O)NC(C)C(C)(C)NC(c2cn(C)nc2C2CC2)=O)CC1 C#CCCC(O)C(=O)NC1C2CC1N(C(=O)C=Cc1cccs1)C2C Cc1ccc([N+](=O)[O-])cc1S(=O)(=O)N1C(C(=O)NC2COCC2O)CC2CC12 c1(-c2nc(C)nn2C2CCC2)c[nH]c2c(Cl)cccc12 Cc1nn(CC(C)C)c(Cl)c1C(N1CCC(NCC2CC2)C1)C C=CC1CCCN(C(C2(C=C)CCN(C(c3cnncc3OC)=O)C2)=O)C1 c1(C(N(CCCNC(c2ccns2)=O)C(C)C)=O)cn(C)cn1 c1(C(N(CCC)Cc2ccc(Cl)cc2)=O)c(Br)nc2n1CCCC2 C1(OC)(CNC(=O)CC2COCCOC2)CCN(C(C2(O)CC2)=O)C1 c1(C(=O)NCCN(CCC)C(c2cc3scnc3[nH]2)=O)ccc2cncn2c1C C1(CNC(=O)CC2CCC2)CCCN(C2CC2)C1 C#CCCC(O)C(=O)NC1CN(C(c2cc(Br)cs2)=O)C1 C#CCCCCCCC(=O)N1CCC(C(=O)NC(c2cnccn2)C)C1 N1(C(C2C(=C)CC2)=O)CC2CCC1CN2C(c1c(C)nn(CCO)c1C(F)F)=O c1(CC(=O)N(C(CNC(c2coc(O)n2)=O)C2CC2)C)cc(F)cc(F)c1 c1(CCC(C)NC(C)CC(C)N)ccccc1F c1(C(=O)NCCC(C)N(C(C(C)c2cncs2)=O)C)cc2cccc(F)c2o1 C(=O)(CC1CNc2ccccc21)NC1CCN(C(C=CC)=O)CC1 C1(C)(NC(CN2CCC(C)(C)C2)=O)CCC(NC(C2COCCO2)=O)CC1 C1(CC(=O)NC(C#C)(C)C2CC2)CN(C(=O)Cc2csnn2)CCC1C C(C(C)(C)CC=C)NC(c1n(CC(=C)C)nnn1)C1CCSCC1 C#CC1CCCCN1C(C1(C)C=CCN1C(C1CCC1C(C)(C)C)=O)=O c1(CC)c(C(N2CC(CNC(=O)CSc3nncn3C)C(C)C2)=O)nnn1CC CC1CC(N=c2nc(C(F)(F)F)[nH]s2)CN1C(=O)C1=CS(=O)(=O)CCC1 c1(NC(C2(C)CCN(Cc3cc(C)c(Cl)nc3)C2)=O)nc2cc(F)ccn2n1 c1(C(=O)NCC23C(CN(C(C(CC)(C)CC)=O)C2)C3)cc2cc[nH]c(=O)c2s1 C1(NC(c2c(CC)cno2)=O)CCCCC1NC(c1cnn(CC(C)C)c1C)=O CCCCC(C)CCC(=O)NCC1CC12CCN(C(=O)C=CC(C)(C)C)CC2 c1(C(N2C(CNC(C(C3CCC3)OC)=O)CCC2)=O)ccc(OC)cc1C(F)F C(=O)(C(O)CSC)N1CC(CC(=O)N(C2(C(=O)OC)CC2)C)C1 n1(CC(C)C)[nH]c(CC(=O)NCC2CC(F)CN2C(C2CCC(=O)O2)=O)cc1=O O=C(CS(=O)C(F)(F)F)N1CCCC1CCCNC(c1ccc(F)cc1)=O c1(OC)ccc(C(N2CCC(C)C(NC(=O)CCCSC(C)C)C2)=O)c(OC)n1 C1(C(N2CCC(N(C(=O)CC=CC(C)(C)C)C)C2)=O)C2CNC(=O)C12 C(CC(CC)C(=O)NC(C)(CSC)C(=O)NCCC1(C)CCOC1)=CC c1(C(=O)NCCN(C)C(C2CCNC(=O)C2)=O)ccnc(OC2CC2)c1 Cc1nn(CC(=O)NCC(C)(CO)NC(=O)Cc2cnc[nH]2)cc1Cl c1(C(C(=O)OC)N(C)CCc2ncc(C)s2)ccc(C)cc1 CC(=O)CCC(=O)N1CC2CC2C1C(=O)NC(CO)CCC1CC1 C(=O)(C1=CCCC1)N1C(C)(CC(N2CCC(OCC)C2)=O)CC1 CC1(COC(C)(C)C)CCC(NC(C2C=CCN(C(=O)OC(C)(C)C)C2)=O)CC1 c1(OC)cc(C(=O)NC2CCCC(CNC(c3cccc(F)c3)=O)C2)cc(C)n1 Cc1cc(C(=O)NCCN(C(=O)C(C)CO)C(C)C)cnn1 Cc1ncc(CC(=O)NC2C=CC(CNC(C3(Br)CC3(F)F)=O)C2)[nH]1 CCC(C)(C)CC(=O)NC(C)(CNC(=O)CCCc1cc(O)ccc1C)C1CC1 C(=O)(CCCC#N)N1C(C)(CC(N2CCC(CC#C)C2)=O)CC1 c1(C(N2CCC(C)(NC(c3ccn(C)n3)=O)C2)=O)ccc2c(c1)CCC=C2 C1(NC(c2c(CC)cncc2)=O)CC2(NC(C3CC=CCC3)=O)COC1C2 O=C(C1=CCOCC1)NCCC1(C(N2CC(O)(C(F)(F)F)C2)=O)CC1 C#CC1CCCN(C(=O)CCC2CC(NC(C3CCCOC3)=O)C2)CC1 c1(CC)nn(C)c(C(=O)NCC2CC(NC(c3cc(OC)ns3)=O)C2)c1Cl CCCC(C)(C)C(=O)NC1CN(c2nnn(C)n2)C1 N1(C(C2CCCC(C)(C)O2)=O)CC(C2CCCCN(C(=O)COCC(F)F)C2)C1 O(NC(=O)CCOC1CC(NC(C2CCCO2)=O)C1)CC(N)=O CC(C)C(C(=O)N1CCCCC(CNC(=O)C(F)(F)C(F)F)CC1)C(C)C C1(c2cn(CCN(CC)CC)nn2)CCN(C(=O)CC2(C)CCCC2)C(C)C1 CC(C)(CCS(C)(=O)=O)NC(c1cc(C(N)=O)cs1)=O C12(C(=O)NC3C(NC(C(C)OC4CCOC4)=O)CC3)CCC(CC1)C2 CCCCC(O)C(C)C(=O)N1CCC(NC(=O)C=CC2CCCN2C)C(C)(C)C1 c1(C(N2CCC3CCC23CNC(C2(Br)CC2)=O)=O)ccc2nncn2c1 CC(O)C(F)(F)C(=O)NC1CC(NC(C2(c3ccccc3F)CC2)=O)C1 c1(NC(c2c(NCc3c(C)ccc(C)c3)c[nH]n2)=O)cccc2c(Cl)ccnc12 c1(C(N2CCC(CNC(C3CC3C(F)(F)F)=O)C2)=O)ccncc1Br c1(C(N2CCC(O)(CC(=O)NCCCCOCC)C2)=O)cc(Cl)ncc1F CC(C)(CCNC(=O)C1=CCCC1)C(=O)NC1CCC(C(N)=O)CC1 CC(C)CCCC(C)NC(=O)N(C1CCN(Cc2cnc(C3CC3)o2)C1)C C1(NC(C2(C3N(C(CCC=C)=O)CCC3)CC2)=O)CCC(C)CC1 c1(C(=O)NC23CC(NC(CCC4N(C)CCCC4)=O)(C2)C3)cc([N+](=O)[O-])cn1C C1(C(=O)NCC2CCCC2NC(c2nc(Cl)oc2C)=O)(OC)CCSCC1 C1(NC(Cc2c(C)ncs2)=O)CCN(C(=O)Cc2cncn2C)CC1F CC(CNC(=O)CCc1ccccc1)C(=O)N(C1CCC1(C)C)C C(C(COC)CC(=O)N(C(C)CCNC(c1cccc(=S)n1O)=O)C)OC C1(C(=O)NCCSCC(=O)N(CC(C)N(C)C)C)CC2(C1)CC(O)C2 CCC(C(=O)N1CCC2CC12C(=O)NCCCN(C)C)C(F)(F)F C1(OC)(CNC(C2CC(C)=NO2)=O)CCN(C(c2ncccc2F)=O)CC1 c1(OC)cc(CC(=O)NC(C2CN(C(C3CCCCC3(C)C)=O)C2)C)ccc1Cl N1(C(c2c(CC)c[nH]c2)=O)CCC(C)C(CC(=O)N(C)CCN2CCCCC2)C1 Cc1cn2cc(C(N3CC(NC(c4cc[nH]n4)=O)CC(F)C3)=O)sc2n1 N1(C(C2CC(=O)NCC2)=O)CC2(C(=O)NCCC(F)(F)F)CCC1CC2 CC(C(=O)N1CC2CC1(CNC(=O)C(C)(C)c1cncnc1)C2)S(N)(=O)=O C1(c2n(CC)nnn2)(Nc2cnc(OC)cc2C(C)C)CCCCC1CC(C)C C(=O)(CCC(C)(C)C)NCC(CCCC)NC(c1ccc(OC2CC2)nc1)=O C1(C(=O)NC2CC(CNC(c3c(CCC)nsc3N)=O)C2)CCOCC1(C)C N1(C(=O)C(F)CC2CC2)CCC(CO)C(Nc2nccc(C(F)F)n2)C1 C1(NC(c2nc(NC(C)=O)sc2)=O)CC(O)CN(C(c2nnc(S)n2C)=O)C1 C1(C(N2CC(NC(Cc3c(C)scc3)=O)C(O)C2)=O)CCCCN1N=O c1(NCc2cnn(C)c2)ccc(C#N)nc1.CCC(C(=O)N(CCO)CC)N(CC)C c1(SC)nc(N(C(c2cc(C)cnc2Cl)=O)CC2(C)CNC2)cc(C(F)(F)F)n1 C(=O)(C(C(C)C)N(C)C)NC(C(C)C)CNC(=O)CCc1cncn1C CC1(C)CC(NC(C2CCOC2(C)C)=O)CN(C(=O)C(F)(F)c2cccnc2)C1 O=NN1CCCCC1C(N1CCOC(CCNC(c2ccc(F)cc2F)=O)C1)=O N1(C(Cc2cn3nc(C)sc3n2)=O)CC(C(=O)NC2CCCCC2)CC2OCCC12 C1(CNC(C(N2CCC(C)(CCO)C2)=O)=O)CC2(C1)CC1(CCC1)C2 c1(C(N2CCCC(CCNC(C3CCC(O)C3)=O)C2)=O)ccc(F)c(Br)c1 N1(c2cc(NCCC(CC)(C)C)ncn2)CCn2ncc([N+](=O)[O-])c2C1 C1(CCC(=O)N(C(C)(C)NCCOC)C)CCCCO1 N1(C(C2(COC)CN(C(C3CCC(=O)NC3)=O)C2)=O)CC(C)(C)C2CCCC12 CC(C)CC(C)(CN=c1ccnc[nH]1)NC(c1cnc(C(C)(C)C)o1)=O CC1Oc2cc(-c3nnc(-c4ccncc4)s3)ccc2N(C)C1=O n1(C(C)C(N2CCC(C)C(NC(C3CCC(C)C3)=O)C2)=O)cnc2ccccc12 N1(C(CC2CN(C(C3(C=C)CCC3)=O)CC23CC3)=O)CCCN(C)CCC1 c1(C(N2CC(n3cc(CCCC(C)=O)nn3)C2)=O)ccc2cnc(C)cc2c1 c1(C(CNC(CSCC)=O)NC(C2CC=CCO2)=O)ccc(F)cc1F N1(C(C2(CC)C=CCC2)=O)CC2(C1)CN(C(=O)CSc1n[nH]c(C)n1)C2 CCC(F)(F)C(C)(C)C(=O)NC1CCCC(CN=c2cc(Cl)nc[nH]2)C1 C(CC(C)(C)C(=O)NCC(C)C(=O)NCC1(O)CCCCC1)SC c1(C(=O)NCCCCCN(C)C(C2(F)CC2)=O)cn(C(F)(F)F)cn1 c1(C(N(C2CC(NC(C(C)c3cc[nH]n3)=O)C2)C)=O)cnc(-c2cccnc2)s1 C1(C(=O)NCC2CCCCCN2C(C23C(=O)C4CC2C3C4)=O)CC2(CCC2)CO1 Cc1ccccc1CC(N1CC=CC1CNC(c1occc1Cl)=O)=O C=C(C)C(C)(C)C(=O)N1CCCC(F)(C(=O)NCC(C)CC(F)(F)F)C1 N1(C(Cc2c(C)scc2)=O)CCCCC(N(C(=O)CC2CCCCO2)C)C1 N1(C(c2c(C#C)cn(C)n2)=O)CC2(CC(C(=O)N(CC(O)CO)CC)CO2)C1 N1(C(CN(C)C2CC2)=O)CCCCCC(NC(c2ccnc(-c3ncc[nH]3)c2)=O)C1 N1(C(c2c(C)cn(C)c2)=O)CC(C)CCC1CNC(=O)Cc1cnns1 CC(CCO)N=c1[nH]c(N2CCCCC(CO)C2)nc2c1COC2 C1(CC(=O)N(CC(CN(C(=O)CC2CC3(CC3)CO2)C)O)C)CC(C)(C)CO1 C1(CC(=O)NC(C(C)(C)OC)C)CCN(C(=O)CC2(C)CC2)CC1 C(CNC(C1(O)CCSC1)=O)(CC(=O)NC(C(O)CO)C1CC1)OC N1(C(C2CC3CCCCN3C2)=O)CC2(C1)CN(C(C1CC3CC3C1)=O)CCO2 C#CC1CN(CC(=O)Nc2ccc(C)cc2Br)CC1O Cc1cccnc1C=CC(N1CCC(NC(=O)CCC2CC2(Cl)Cl)CC1C)=O C(=O)(C1=NN(C)C(=O)CC1)NCC(=O)N(CCCCC)CCc1cncnc1 C=CCCCCC(=O)N1CC2CC1CN2C(c1cc(CC)[nH]n1)=O c1(COCC)cccc(CNC(=O)CC(O)Cn2cc(-c3cn[nH]c3)nn2)c1 C#CCCCCCCCC(=O)N1CC(O)(C(C)NC(=O)C(C)CC)C1 Cc1cccnc1CC(=O)N(C1CN(C(c2c(CO)noc2C)=O)CC1F)C S(=O)(=O)(c1c(C)cccc1Cl)N1CC(N(C(C)=O)C)C1 n1(CC)cc(C=c2sc(=C(C#N)C(=O)c3nccs3)n(C3CC3)c2=O)cn1 c1(C(=O)NC(CC)CNC(=O)C(C)n2cncn2)cccc(C(F)(F)F)n1 n1(CC)c(C)nn(CC(N2CCC(CCOC)(NC(=O)C3=C(Cl)CC3)C2)=O)c1=O CCS(=O)(=O)CC(=O)NCC12CCC1CCN2C(c1cscc1C)=O C(=O)(C1=CCCSC1)N1CC(CCCCNC(CC2(C=C)CCC2)=O)C1 C12(C(N(CC(C)(C)NC(c3ccnn3C3CC3)=O)C)=O)CCC(C(F)F)(CC1)C2 C12(CC(=O)N(C(CCNC(c3n(CC)ncn3)=O)C)C)CCC(CC1)CC2 Cc1ncnc(O)c1C(=O)NC1CC2CC(NC(C3(C(F)(F)F)CC3)=O)C2C1 Cc1cccc(-n2cc(-c3ccccc3C(=O)NCC3(CF)CC3)nn2)c1Br N1(C(c2c[nH]c(=N)o2)=O)CC(=O)N2CCOCC2(CNC(=O)COC(F)(F)F)C1 CC(CN(C)C)CCC(=O)N1CC(CN(C)C(C2CC(CF)C2)=O)C2(CC2)C1 C1(N(C(C(C2CCC2)OCC)=O)C)CCC(NC(C2CC(F)C2)=O)CC1 N1(C(=O)C(F)Cc2ccccc2)CCN(C(c2cnc(Cl)s2)=O)C(CCO)C1 c1(C(N2CC=CC(NC(Cc3nnn(C(C)(C)C)n3)=O)C2)=O)ccc(=O)n(O)c1 CC(C)CC(O)CC(=O)NCCOc1ccn(C)n1 C(C)(C)(CCCCC(=O)N1CCN(C(=O)CC2=CCCC2)C(C)C1C)OC C1(NC(CCC(C)(C)NC(=O)C2=CCCCC2)=O)CCCCCCC1O C1(C(N(CCC(C)NC(CCOCC)=O)C)=O)Cc2cc(C)ccc2S1 c1(C(N2CC(O)(CNC(c3cccc(C)c3F)=O)C2)=O)cnc2c(F)cccn12 CCC(C(=O)NC1CC(CCNC(c2cnc(C(F)(F)F)nc2)=O)C1)C(C)O C1(CC(=O)N(CCCNC(CCC(C)C)=O)CCO)CC(=O)NC(=O)C1 N1(C(c2nc(CS(C)(=O)=O)sc2)=O)CCN(C(=O)C#CC(C)(C)C)C(C(F)F)C1 C1(NC(C2CCCS2)=O)CC2CCC1CN(C(c1nccc3c1NCCC3)=O)C2 N1(C(c2c(C(C)=O)cn(C)n2)=O)CC2CC(NC(C3CC3(F)F)=O)C2C1 c1(C(=O)NC(C)CNC(c2occc2-c2ccccc2)=O)ccnc2[nH]nnc12 Cc1cc(CC(=O)NC2(CCNC(=O)CCNCC)CC2)sn1.C1(C=O)CC1C c1(C(c2n(CCCC)nnn2)NCCS(=O)(=O)N(C)C)ccc(C)nc1 N1(C(C(C2CCCC2)OC)=O)CCC(CNC(C2CN(C)C2)=O)C(O)C1 N1(C(C2CCN(C)C2=O)=O)CC2(CCN(C(C3CC3c3ccco3)=O)CC2)C1 C(C)(C)(CC(=O)NCC(C1CCN(C(=O)C(F)=C2CCCC2)CC1)C)OC N1(C(c2cc(CC)nn2C)=O)CC(NC(C2CCCC2(F)F)=O)C2CCCC2C1 N1(C(c2ccnc(OC)n2)=O)CC2CN(C(c3c(Cl)csc3Cl)=O)CC2C1 c1(CCN2CCN(c3nccc(C(=O)OC)c3C)CC2)ccc2cnccc2c1 c1(C(N2CC(NC(C(C)c3ccsc3)=O)C(C)C2)=O)ccc(N)c(Cl)c1 c1(C(=O)NC2C(NC(C3CN(C(C)C)C(=O)C3)=O)CCC2)ccc2cc[nH]c2n1 c1(C(=O)NCCN(C(=O)CN2CCC(O)CC2)CC)nc(=N)cc[nH]1 C(C)(CN=c1[nH]c(N2CCC(CS(N)(=O)=O)C2)nc(=N)[nH]1)(C1CCOCC1)OC CCCCCCC(C)NC(=NCCc1ccc(Cl)cc1Cl)NCc1[nH]nnc1C C#CCC(C)(C(=O)N1CCC(O)(C(N)=O)C1)NC(c1[nH]nnc1CC)=O C1(NC(CSCC(=O)OC)=O)CCN(C(C2(C(C)(C)C)CCC2)=O)CC1 C(=O)(C1Cc2ccccc21)NC(CN(C(C(C=CC)O)=O)C)(C)C C=C(C)CC(C)C(=O)NC(C1CCCCC1)CNC(=O)Cc1ccc(CC)nc1 N1(C(C2N(C(CC3(C(=C)F)CCC3)=O)CC=CC2)=O)CC2(C1)CC(C)(C)C2 c1(C(N2CC(CNC(CC(=O)NCC)=O)C3C2C3)=O)ccc2nc(S)[nH]c2c1 n1(C(C)C)cnc(CNC(c2coc(CNC(=O)C(C3CCCCC3)C)c2)=O)n1 NS(=O)(=O)CCCCOC(c1nn(CC(F)(F)F)cc1Cl)=O c1(OC)ccc(C=CC(=O)NC2CN(Cc3ccccc3)CC2C)cc1OC c1(CC)c(C(=O)NCCOC2CCN(C(=O)C(O)C3CC3)CC2)nnn1CC C(=O)(C(O)CC(C)C)N1CCC(O)(CCNC(c2c(C)n(C3CC3)cc2)=O)C1 N1(C(C(CC)n2cccn2)=O)CC2CC1C2NC(=O)C=CC1CCOCC1 C(=O)(C1=Cc2ccccc2OC1)NCCC1N(C(C(CC)C)=O)CCCC1C N1(C(c2c(C)nc(O)[nH]2)=O)CCOC2(CCN(C(=O)CC3C=CS(=O)(=O)C3)C2)C1 Cc1ccc(F)c(CNCC23CCC(NC(=O)C(O)c4ccsc4)(CO2)C3)c1 c12ccc(cc1)c(=O)n2C(=O)CCN1CCC1CC(=O)O.S(C)(=O)(=O)CC C12(C(=O)NCc3c(CCNC(C4C(C(C)(C)C)C4)=O)ocn3)CCCC1C2(F)F c1(CCC(=O)NCC2CCC2NC(C2(c3cccs3)CC2)=O)ccc2ncsc2c1 C#CCC(C(=O)N1CCC(CC(C)(C)C)C1)NC(=O)C(C(C)O)N(C)C CC1CC=C(C(=O)NC2(CO)CCN(C(c3cnc(N(C)C)nc3)=O)C2)CC1 c1(-c2n(CC)ccn2)cc2ccccc2nc1C(=O)NCC1CCC(CC)CC1 C(C)(CC(=O)N(C1(C)CC1C(F)(F)F)C)NC(C=CC)=O c1(C(=O)NC(CNC(CNc2cc(C)oc2C)=O)C)cc(Cl)ccc1C(C)C c1(C(N(CC(C)(C)CNC(=O)C(=O)NC2CC2)CC)=O)cc(OC)c(C)c(OC)c1 N1(C(c2cc(C)n(C3CC3)c2C)=O)CCCCCC(NC(=O)C(F)C(F)(F)F)C1 C(c1ccc2c(c1)CCO2)=CC(=O)NCC(CN(C(c1ncc(C)cn1)=O)C)C c1(CNC(CCN(C(C=CCC)=O)CCO)=O)ncnn1C1CC1 c1(C(=O)NC2C=CC(C(=O)Nc3ccc(C)cn3)C2)cc(F)cnc1Cl N1(C(C(c2cn(C)nc2)(C)C)=O)CCN(C(C2CC2F)=O)C(CO)C1 O=C(C1=CC2C=CC1C2)NCc1ocnc1C(=O)NC1CCCC1(F)F n1(CC(=O)NCC2(NC(CC(C)(C)O)=O)CCOC2)cnc2c1CCCC2 c1(COC)cncc(C(=O)N(C2CC(NC(c3cc(Cl)cnn3)=O)C2)C)c1 C12(NC(C(C)n3cncn3)=O)CC1CN(C(=O)CC(=O)OCCC(C)C)C2 N1(C(CCCCNC(C2=NOC(C)C2)=O)=O)CCC2(CCOC2=O)C1 Cc1cc(C)c(CC(=O)NCC(CNC(=O)C(C)C2CC2)C(F)(F)F)c(C)c1 Cn1ncc(C(=O)NC2(CCNC(c3cn(C(F)(F)CO)nn3)=O)CC2)c1C#N C1(CC=C)(NC(=O)CC(c2cccs2)NC(N)=O)CCN(C(=O)C=CC2CC2)C1 c1(C(=O)OC)cc(Br)ccc1C(=O)C(c1cncnc1)C Cc1ccc(C=CC(=O)NC23CC(C(N4CC5(C)CC4(CO)C5)=O)(C2)C3)cc1 N1(C(c2c(O)nnc(C)c2C)=O)CC2CCC(NC(=O)Cc3cccs3)CC2C1 c1(C(=O)NCCN(C(=O)Cc2cnnn2C)CC)ccc2nc(O)[nH]c2c1 C1(CNC(c2c(OC(C)C)cccc2)=O)CC2(C1)CN(C(C1CS(=O)(=O)C1)=O)C2 c1(CS(C)=O)c(C(=O)OCC(C2CCC(F)(F)CC2)=O)oc2ccccc12 N1(C(C(C(CC)O)C)=O)CC2CCCN(C(=O)CSc3cccc(F)c3)C2C1 CC12CC(C(=O)NC3CC3CNC(c3nc(C4CC4)cs3)=O)(CCO1)C2 c1(NCCNC(=O)CCC2CCC2)cc2c(C(=O)O)cccc2s1 c1(CNC(CCC2N(C(C3CCN(C)CC3)=O)CCC2)=O)ccc2ocnc2c1 O=C(N=c1[nH]oc2cccnc12)C1CN(Cc2ccc(F)c(Br)c2F)CCO1 c1(C(N(C2CCN(C(=O)Cc3nc(C)sc3C)C2)CC)=O)csc(=NC)[nH]1 N1(C(CCCC(N)=O)=O)CCCCC2(CCN(C(=O)CCN3CCCC3=O)C2)C1 c1(C(N2CC(N(C)C(C34CCC3C4)=O)C(O)C2)=O)ccc(Br)cc1F c12ccc(Cl)c(c1)NC2=O.C1(NC(CC2(NC(C)=O)CC2)=O)CC(C2CC2)C1 c1(C(=O)NCCC2CCC(NC(CSc3n(C)ncc3)=O)C2)cc(N)ccn1 c1(CN(C(=O)NC(c2cc(OC)ccc2F)C)CC)oc2ccccc2c1CO c1(C(N2CC(NC(C(CC=C)(F)F)=O)C(OC)C2)=O)cc(S(=O)(=O)NC)cn1C C1(C)(OC)CCN(C(C2(NC(c3ccc(C#N)s3)=O)CC2C)=O)CC1 c1(OCC)ccc(C=CC(=O)NCC2CCN(C)C2C)cc1C C(C(C)(C)CC(C)NC(C1(CSc2cccc(Cl)c2)CC1)=O)OC N1(C(CN(CC)CC)=O)CC2(CCN(C(C3CC4C=CC3C43CC3)=O)C2)C1 N1(CC)N=C(C(=O)N2CC(N(C(=O)CCCC3CCCC(=O)N3)C)C2)CCC1=O N1(C(=O)NCC(c2ccc(F)cc2)(F)F)CC2C(C(F)(F)F)CC2(C(=O)O)C1 N1(C(CNC(CCC(C)C)=O)=O)CC2CCCC2(NC(C23CC(C)(C2)OC3C)=O)C1 CC1(C)CC(NC(=O)COCC2CCOCC2)CN(C(c2cncc(N)n2)=O)C1 CCCC(CNC(=O)C(C1CCN(C(C2(n3cccn3)CC2)=O)C1)C)CCC c1(OC)nccc(CNC(C2CCC2CNC(=O)CC2(O)CCOC2)=O)n1 N1(c2n(CCC3CC(C)(C)OCC3)nnn2)C(CO)CC2CCCCC12 C1(C(N(CCNC(c2ncn(C(C)C)n2)=O)C2CC2)=O)CCCC12OCCO2 CC1(C)CCCC(CC(=O)NC23CC(C2)N(C(c2cccc(Cl)c2Cl)=O)C3)C1 C(CCCCCNC(c1cn(C2CCC2)nn1)=O)N(C(CCN(CCC)C)=O)C C1C(CC2CC2)C(=O)N(C(C)COC(C)C)CC(=O)N1.C(CCC)SCC=C c1(N(c2cccc(OC(C)C)c2C)CC2(C)CN(CC)C2=O)cccc(Cl)c1C C1(CNC(C(C(C)C)C)=O)CN(C(=O)CCNC(C2CCC2)=O)C(C)(C)C1 C(=O)(C(C)(C)C(=O)NCC(C)(C)CN(C(=O)C(O)CSC)C)OC c1(SCc2nc(Cc3n(C(C)(C)C)cnc3)on2)cccc(S(C)(=O)=O)c1 c1(C(N2C3CC(NC(C4CCCCC4)=O)(C3)C2)=O)ccc2ccoc2c1 C1(NC(c2cc(C(F)F)[nH]n2)=O)CC2(C1)CN(C(c1coc(Br)n1)=O)C2 C1(C(=O)NC2CCC(NC(c3cn(C(C)(C)C)nn3)=O)C2)CC2CC1CO2 C12(NC(C(C)OCC(C)C)=O)CCCN(C(C3C(C)OC(C)C3C)=O)CC1C2 CCCC(CC)C(=O)NC1CN(C(c2sccc2F)=O)C(C)(C)C1 N1(C(C(C)(C)C)=O)CC(CN=c2[nH]nco2)C(C)(C)C1 C#CCC(C(=O)NOCC)NC(=O)CCCCCC c1(C(=O)NCC2(OC)CN(C(c3cc(C)n(C)n3)=O)C2)c(N)cc(Cl)cc1F Cc1sc(N)c(C(N2CC3CCC3(CCNC(=O)C3=C(Cl)CC3)C2)=O)c1C N1(C(C(CC)C#N)=O)CCC(N=[N+]=[N-])(C(=O)Nc2cccc(C)c2C)C1 C1(C)(C(N(CC(C)NC(C2(C)CCC(=O)C2)=O)C)=O)CCS(=O)(=O)CC1 N1(C(C(C(C)(C)O)F)=O)C(C(=O)NC2COC(C(F)F)C2)C2CC(O)C1C2 c1(CC)nn(C)c(CC)c1CC(N1CCCC1)=O.C12(CCOCC1)C(=O)N2.C(C)(C)O CCCCC(C)(F)C(=O)N1CCC(C2CC2)(NC(C2CCSCC2)=O)C1 CC1CCC(NC(c2cc(Br)co2)=O)CN1C(c1ccccc1SCCO)=O c1(C(=O)NCc2cccc(Cl)c2)n[nH]c2ccc(-c3ccnn3C3COC3)cc12 c1(C(C(=O)NCC2N(C(CCOC(C)C)=O)CCCC2)O)ccc(Cl)c(Cl)c1 c1(NS(C)(=O)=O)cccc(NC(C2C=CCCC2C(F)(F)F)=O)c1 Cc1nc(C)n(CC(=O)N(C(C)CN(C)C(C2(Nc3ccccc3)CC2)=O)C)n1 c1(CC(=O)OC)ccc(S(=O)(=O)CCN(CC(CN(C(CC=C)=O)C)O)C)cc1 C1(CNC(C(C(C)(F)F)F)=O)CN(C(c2ncoc2C2CC2)=O)CCC1(C)C c1(CSCCNC(c2cccc(F)c2F)=O)cc(F)ccc1Br c1(C(=O)NCC(CC)NC(C2(C)COCC2(F)F)=O)cc2n(n1)CCCC2 Cn1nc(CC(=O)NC2CC(CCNC(=O)CC3CCCO3)C2)cc1C(F)(F)F C1(NC(C(CC=C)CC)=O)CC1C1CCN(C(c2cnc[nH]c2=N)=O)CC1 C1(CCOC)(NC(=O)CCCn2cccn2)CCN(C(c2cc(C)on2)=O)C1 C(=O)(C1=C(C)CCCC1)NC1(COC)CCN(C(=O)Cc2cccc(SC)c2)C1 C(=O)(CCCCNC(=O)COc1ccn(C)n1)N1C(C)CCC1 C1(C(C)(C)C)(CNC(c2occc2C2CC2)=O)CCN(C(C2CCSCC2)=O)C1 CC(CC(F)F)C(=O)NCCN(C(=O)COCc1ccnc(O)c1)C1CC1 c1(C(N(C2CCCN(C(C(C)SC)=O)C2)C)=O)cc(C)cc([N+](=O)[O-])c1N N1(C(C2CSCCS2)=O)CC2C(CNC(C3(CC4CC4)CC3)=O)C2C1 C1(CNC(c2c(C)cco2)=O)CC12CCN(C(=O)CC1(C)CCS(=O)(=O)N1)CC2 c1(C(N2C(C)C(NC(C3C4CC5C(C4=O)C35)=O)CCC2)=O)cnc2n1CCOC2 N1(Cc2noc(C)c2Br)CC(C(=O)OC(C)(C)C)C(S(C)(=O)=O)C1 c1(C(=O)NCCNC(C=CC)=O)ccc(NC=O)cc1.C1C(C)(C)N1 N1(C(C2C(CNC)CCC2)=O)CCC(c2nccn2C)CC1 c1(N2CC2)cc(C(N)=O)nc(Cl)n1.N1(C(CSC)=O)CCCCCC1.C1(=O)C(C)N1 c1(C(N2CCC(NC(=O)Cn3cccn3)(CO)C2)=O)ccc(Cl)c(F)c1F N1(C(C(C)=C2CCCC2)=O)CCCC2(CC(NC(=O)C3Cc4ccccc43)C2)C1 c1(C(=O)NC(CC(C)NC(c2n(C(C)C)ncc2)=O)C)cccn2nnnc12 CC1=C(CNC(=O)C(C2CCN(C(=O)C(=O)C3CCCC3)C2)F)CCC1 C1(CNC(CC(C)SC)=O)CC(F)CN1C(=O)C(C)NC(c1cccs1)=O N1(C(C(COC)C)=O)CC(CNC(=O)COCC(=O)OC(C)(C)C)C(O)C1 N1(C(CC=CC=C)=O)CC(NC(c2conc2C(C)(C)C)=O)CCC1C C1(CNC(c2c(C)nco2)=O)CCCC12CCN(C(c1ccsc1C#N)=O)CC2 C(C)(CO)(CN=c1ccnc(N2CCCC(CC(F)F)C2)[nH]1)OC Cc1cc(Cl)ccc1NNC(=O)C=Cc1ccc(F)cc1F C1(C(C)O)CCC(NC(=O)CCC2CCCN2C(c2cnco2)=O)CC1 Cc1ccc(C(=O)NCCC(=O)NCCC[Si](C)(C)C)cc1F C1(CNC(c2ccc(F)cc2)=O)CCCN(C(c2sccc2CO)=O)CC1 C(=O)(C1CCCc2c1ncn2C)NCC(C)NC(c1cc(C#C)cc(F)c1)=O C(c1ccncc1)=C(C)C(=O)NCC(C)CNC(=O)COCC1CCOC1 c1(C(N2CCC(NC(Cc3ccn(CC)n3)=O)CC2)=O)ccc(Cl)cc1C c1(C(N(C2CN(C(C(Cn3ccc(C)n3)C)=O)C2)C)=O)ccc(=O)n2c1CCC2 C1(NCCC(CC2(CO)CCOCC2)O)CCC(F)(F)CC1 c1(C(N2C(CN(C)C(C3(CO)CCCO3)=O)CC(F)C2)=O)cncc(Cl)c1Cl CC(=O)C(C)CC(C)C(=O)NCc1ccc(C(=O)NCC2(CCO)CC2)o1 CCCC(C)(O)C(=O)N1CCN(C2CCCN(C(=O)C(C)NC(N)=O)C2)CC1 C1(C2CCCCC2)(NC(C2N(C(C(CC)Cl)=O)CC(O)C2)=O)CC1 C#CCC(CC(=O)NC(CC)C(C)(C)O)NC(=O)C(C)OCC(C)C c1(C(C)C)ccc(C(=O)NCCC(O)CNC(C2CCCC2F)=O)cn1 c1(CC(=O)NC(CCOC)CNC(=O)Cc2ccco2)ccc(F)c(F)c1 CCC(CC)CCCC(=O)N1CC(CNC(=O)CSc2nncn2C)C2CC12 C1(CNCCN(C(=O)C(F)OC(F)(F)F)Cc2cccc(Cl)c2)COCCOC1 c1(C(=O)NC2(CCC(=O)NC3CC(C#N)C3)CCC2)ccc2c[nH]nc2c1 N1(C(c2c(CNC(Cc3ccc(C)nc3)=O)ccs2)=O)CCC2C(O)C(C)(C)C12 c1(CC)ncc(C(=O)NCC(C)(CNC(c2ccccc2OC)=O)OC)cn1 N1(C(CC(CC=C)(C)C)=O)C2CCC1C(F)C(NC(=O)C(F)C(C)(F)F)C2 C1(CC(N2C(CC(=O)NC(C(=O)OCC)C3CC3)CCC2)=O)CCC(=O)NC1 c1(C(=O)NC2C(NC(c3csc(Cl)c3)=O)C2)ccccc1Nc1ccccc1 N1(C(C(CCC)O)=O)CCC(CNC(c2cccnc2OC(F)F)=O)C(C)C1 N1(C(C(C)NC(=O)C2CC2)=O)CCC(CN(C)C(c2cccc(=O)o2)=O)CC1 C1(C)(C(=O)NCC2(NC(C3CCC(CC)O3)=O)CCC2)CC(C#N)C1 C(c1cnc2ccccc2n1)=CC(=O)NC(C)CCNC(C1(Cl)CC1)=O Cc1cc(C(=O)NC2CC2NC(C2(C#N)CC3CC3C2)=O)cc(C(F)F)c1 c1(NC(=O)NC(c2ccc(C)nc2)C2CC2)c(-c2ccccc2)nc2ncccn12 n1(CC(=O)NCC2(N(S(=O)(=O)C3CC3)CCO)CC2)c(=O)sc2cc(Br)ccc12 C(=O)(CC(C)C(=O)N1CC2CC2(CNC(C2CCC2(F)F)=O)C1)OCC c1(C(=O)OC(C(C)OCC=C)C)cnn2c(C(F)F)cc(C)nc12 c1(C(N2C(CNC(CCC(=O)NCCC)=O)CC2)=O)cc2cc(F)ccc2cn1 N1(C(C(C(C)C)SCC)=O)CCCC(C(N2CCC(OC(C)=O)C2)=O)C1CC C1(C(=O)NCCNC(=O)CS(=O)(=O)C2CC2)COc2ccc(O)cc2O1 c1(C(N(CC(CN(C(CSCC=C)=O)C)O)C)=O)sc2nc(C)nc(C)c2c1C N(C1COc2cc(Br)ccc21)C(C(=O)Nc1cccc(SC)n1)=O C1(OC)CC(NC(C2OCCC2C)=O)CN(C(c2csnn2)=O)C1 N1(C(c2ncn(C)c2)=O)CC2CCC1C(CNC(C1(C)CCC(=O)NC1)=O)C2 C=CCCCC(=O)NC1CC1NC(c1cn(CC(N)=O)nn1)=O c1(C(=O)NC2CCCCC2)noc2c1CN(CC(=O)Nc1cc[nH]n1)CC2 C1(C(=O)NCCCCC2CN(C(C3C(C)CC(C)O3)=O)C2)CC(=O)NC(=O)C1 C#CC1(C(=O)NCc2cncc(C(=O)NC3C=CCCC3)c2)CC(=O)C1 C1(NC(CCSCC)=O)C2CN(C(C3(C)COC(=O)C3)=O)CC12 Cc1ccc(S(C)(=O)=O)cc1C(=O)NCC1=NOC2C3CCC(C3)C12 CCC(CC)C(C)C(=O)NCC12CCC(CC1)N2C(=O)C(F)=C1CCC1 C(=O)(C(C#N)C(C)(C)C)NCc1cc(C(N2C(C(CC)O)CCCC2)=O)ncc1 CCCCS(=O)(=O)NC(C1(C)CCN1C(=O)NC(=O)C(Cl)(Cl)Cl)=O C1(NC(C2CCC(C)(CC)O2)=O)CC2CCC(C1)N2C(C1CCC2CC2C1)=O Cc1cc(Cl)nc(Cl)c1CNC1CC(CC(=O)Nc2cnccc2C(N)=O)C1 C=CCCC(C)(C)C(=O)NC1CCC1NC(=O)Cc1ccn(C(C)C)n1 c1(NC(CC)CN(C(=O)COCc2ccccc2)CC)ccnc2ncnn12 C1(C(C)=O)CC(CC(=O)NCC(C)(C)NC(c2ccccc2CC#N)=O)C1(C)C S(=O)(=O)(c1ccccc1)N1CC(C(C)NC(=O)NC2CCOC(C)(C)C2)OCC1 c1(C(N(C)CC2CCN(C(C3CC(C)(C)O3)=O)C2)=O)ccc(F)c(C(F)(F)F)c1 C1(CC(=O)Nc2ncccc2I)CCC(NC(c2ccnnc2)=O)CC1 N1(C(c2cncc(C)n2)=O)CCC(C)C(NC(C2CCC(=O)N2C(C)C)=O)C1 C12(NC(c3cnc(Cl)s3)=O)CCCC1CN(C(=O)Cn1ncc3ccccc13)C2 C1(NC(C(Br)=C(C)C)=O)CN(C(c2ccc(F)cc2F)=O)C2CCCCC12 c1(C(=O)NC(CCNC(CC2(C=C)CCC2)=O)C)ccc(C2CCCC2)cc1 N1(C(c2scc(C)c2)=O)CC(NC(c2cnc(Cl)cc2N)=O)CCC1C c1(C(N(CCOC)CCNC(c2ncc(C(F)F)s2)=O)=O)cccc(C(C)C)c1 CCCCC(O)C(C)C(=O)NCc1cnn(C)c1C(=O)NOCc1ccccc1F C1(NC(CCCCN(C(C2OCCN(C)C2)=O)C)=O)CCCC(F)(F)C1 C1(C2CCOCC2)(C(N(C(C)CNC(c2cnc(C#N)s2)=O)C)=O)CC1 C(CCC(C)C(=O)NCc1cc(C(=O)NC2CC3(CC3)C2)ccn1)OC C(c1cn[nH]c1)=C(C)C(=O)N(CCC(C)NC(=O)C=CCO)C N1(C(C2(CC)CCNC2=O)=O)CC2CCC(C1)N2C(C1(C)CC=C(C)CC1)=O Cc1nccc(C(=O)NCc2ccc(C(N3CCC4CC4C3)=O)s2)c1N c1(CC(=O)NC2CC(CNC(C(COC)(C)O)=O)C2)c(C)nn(CC(C)C)c1C N1(C(C2C(C)C2C)=O)CC2CCN(C(c3cc([N+](=O)[O-])n[nH]3)=O)CC2C1 c1(C(N(C2CCN(C(=O)COCC3CCC3)C2)CC)=O)n[nH]c(C)c1C C(C(=O)NC(c1ccccc1F)CNC(c1cnc(C2CC2)[nH]1)=O)(C(C)C)OC C1(NC(c2c(-c3c(OC)cccc3)onc2)=O)CCNC12CCCC2 CC1(F)CC(C(=O)N(CCCNC(=O)CC2CCCO2)CC2CCCCC2)C1 c1(CC(N2CC(C)C(NC(C3CN4CCC3CC4)=O)C2)=O)cccc2[nH]ncc12 C1(CNC(c2ccn(CCF)n2)=O)CCC(=O)N1.C12(CC1)C(C)NC2=O c1(NC(C)C(=O)OC(C)(C)C)cc([N+](=O)[O-])cnc1Br C1(CNC(CN(CC(C)C)C(c2ccc(CC)[nH]2)=O)=O)(CC)CC(C)(C)C1 N1(C(C2=CC(C)C2)=O)CC(CO)C2(C1)CN(C(C1(C(=O)NC3CC3)CC1)=O)C2 c1(C(N2CCC(C)(NC(=O)CC3CCOCC3)C2)=O)cnc2c(c1)CNC(=O)N2 C=CCC(F)(F)C(=O)N1CCC(NC(C2(NC(=O)OC(C)(C)C)CC2)=O)C(C)C1 C1(CC)C(NC(c2cnco2)=O)CCN1C(=O)CCOCC(C)C C1(NC(c2cc(CNC(c3c(CC)ncnc3)=O)[nH]n2)=O)CCc2nncn2C1 C(=O)(C1=CC2CC(C1)CC2O)NCC(CCCC)NC(c1[nH]cc(C)c1C)=O c1(N2CCC(NC(C3CCC4(CCC4)CO3)=O)C(F)C2)ncnc2c1CCC2 CCCCCC(CC)C(=O)NCCN1CCN(C(=O)C=CC(=O)NC2CC2)CC1 c1(C(=O)NCC2OCCC(NC(CCOC)=O)C2)cnn2cc[nH]c(=O)c12 N1(C(c2cn(CC=C)nc2)=O)CCCCC1CN(C(=O)CC(C)c1ccco1)C N1(C(c2c(CC)n[nH]c2)=O)CCC2CCCC(C1)N2C(=O)Cc1cc(C)sc1C CC(CCC(=O)NC1CCN(C(c2cc(C3CC3)nn2C)=O)C1C1CC1)N(C)C C1(S(C)=O)(CNC2(c3nnnn3C(C)C)CC(CCCC)C2)CCC1 C(N=c1nc2ncccn2[nH]1)c1nccc(-c2ccc(S(N)(=O)=O)s2)c1 c1(C(C)=O)ccccc1Oc1cnc(-n2cccn2)cn1.C12CCN(C1)C2=O C1(C(=O)NCC23CC(NC(C(CCC)OC)=O)(C2)C3)CC2CC2CC1C c1(N2CC(C(=O)Nc3ccc(C)nc3CO)C(O)CC2)ccnc2ccnn12 N1(C(N2CCC(C)(CSC)CC2)=O)CCSC2CCCCC12 N1(C(c2cc(C)cc(Br)c2)=O)CC2CN(C(=O)C=Cc3ccc(O)cc3)CC2C1 c1(C(N2C(C)CC(NC(=O)C=CC3CCCCC3)C2)=O)cc(F)cc2nn[nH]c12 n1(CCOCC)nnnc1C(C(C)(c1ccccc1)OC)NC(C)(C)COC N1(C(CC2N(C)CCC2)=O)CC2C(CNC(=O)C=CCN3CCCC3)C2C1 CC1=C(C(=O)N(C2CN(C(c3nonc3N)=O)C2)C)C=C2CCCN=C2N1 N1(C(C(C=C)(C)C)=O)CC2CC(CNC(C3CC3c3ccncc3)=O)C2C1 N1(C(c2ncc(CC)cn2)C(=O)NCCSC)CC2CCCC2(CN(C)C)C1 CC(CC(=O)NCCNC(c1ccc(C(C)(C)C)s1)=O)C1CCCCC1 C=CC1(CC(N2CCC(C)C(NC(C34CC3COC4(C)C)=O)C2)=O)CCCCC1 C(=O)(C=C1SCC(=O)N1C)NC1(COC)CCN(C(c2cnc(CCC)s2)=O)C1 CC(C)(C(=O)N1CCC(CSC2CC2)C1)ONC(c1coc(C(N)=O)c1)=O C(CCS(C)=O)(C(=O)NCC(C1CC1)NC(=O)CCCc1cccs1)N(C)C C1(NC(C=C(COC)C)=O)CCC1C(=O)NC(c1cscn1)CO C(CCO)(C(C)(C)C)NC(C1CC(NC(CC2CCN(C)C2)=O)C(O)C1)=O C=CCC(C(=O)NC1(C(=O)NC(CC)C(C)(C)O)CCCCC1)OC N1(C(C2(OC)CN(C(c3ccc(SC)o3)=O)C2)=O)CCC(C(C)(C)O)CC1 c1(OCC)ccc(C(=O)NC2(C(C)NC(C3CN(S(C)(=O)=O)C3)=O)CC2)cn1 c1(SC)nc(C)c(CCC(=O)NC2(CCCNC(C3(C)CC3F)=O)CC2)c(O)n1 c1(C(N2CC(F)(C(=O)NC(CC#C)(C)C)C2)=O)ccc(O)nn1 N1(C(CN(C(C)C)C)=O)CCN(C(c2cc(-c3ccn(C)n3)on2)=O)CC1CO S(=O)(=O)(c1cc(F)ccc1F)N1CC2CN(C(=O)CCc3ccccc3F)C2C1 CCC(C)(CN(C(=O)CCNC(=O)Cc1cn(C)cn1)C)OC N#CC1(CC(N2CCC(NC(C3(CCS(N)(=O)=O)CCC3)=O)CC2)=O)CCOC1 Cc1oc(C(N2CCC2CNC(c2ccc(CO)cc2)=O)=O)cc1S(C)(=O)=O c1(C(=O)NC(C(C)C)CCNC(=O)C(C2CCCCC2)=O)ccc2ccnn2c1 N1(C(C2C(C)CC2)=O)CCCC(CNC(c2csnn2)=O)C1 c12ncc(cn1)c(=O)[nH]2.c1(N(C2CCN(CC)C2)C)nccc(C(F)F)n1 c1(C(=O)NC2CN(C(Cc3ccc(C)nc3)=O)CC2C)ccc(C(C)C)nc1O C1(C(=O)NOCc2ccncn2)(NC(C(C2CCCCC2)C)=O)CCN(C)C1 C=CCCCCCCCC(=O)Nc1cccc(NC(C)=O)c1C C1(C(=O)NCCCN(C(C2COC3CC2C3)=O)CC)CNC(=O)CC1C(F)(F)F C(C(C(=O)N(C)Cc1cnn(C)c1)NC(=O)CCn1ccnc1C)OCC C1(OC)CN(C(=O)C(C2CCCC2)NC(C)=O)CC1NC(c1ccc(=O)oc1)=O c1(C(N2C3CN(C(C(CC=C)(C)C)=O)C(C3)C2)=O)c(Cl)sc2nnsc12 C1(NC(COCc2n(C)cnc2)=O)CCC2CN(CCc3ccccc3)CC2C1 C1(CCC)CCCN(C(C2CCN(C(c3cncc(C)n3)=O)C2)=O)C1 C1(C(N2CCC(OCc3cn(C)nn3)C2)=O)CC2(CCC(N)CC2)C1 c1(C(N2CC(N(C(=O)CSC(C)(C)C)C)C(F)C2)=O)csc2ccccc12 c1(C(=O)NCC(CCCC)NC(=O)Cn2nnc(=O)[nH]2)cc[nH]c2nccc1-2 CC1=CC=CNC(=O)C(=O)NC(C)C1CCN1CC(OCCCO)CC1=O C1(CNC(c2c(CC)c[nH]n2)=O)CCC2COCCC2C1 CCC(C)(CC)C(=O)N1CCN(CCN(C)C(C2(CC(C)C)CCC2)=O)CC1 N1(C(C(CCOC)C)=O)CC(NC(=O)C2=CSCS2)CC(F)C1 c1(C(N(CCCCN(C(=O)CC2CC3CC3C2)C)C)=O)csc(O)n1 N1(C(CC(CCC)CC)=O)CCN(C(c2cccc(CCO)c2)=O)CC12CCC2 N1(C(=O)C(N2CCN(C(c3ccccc3)CO)CC2)=O)CCCC(C(=O)O)C1 C1(C(=O)NCc2occ(C(N(C)Cc3ccncc3F)=O)n2)CC2C=CC1CC2 N1(C(CC(C)(C)F)=O)CC2CC2(CNC(c2ccnc(NC(C)C)c2)=O)C1 c1(NCC2C(NC(C34CCC(F)(CC3)C4)=O)CCC2)ccc([N+](=O)[O-])cn1 C(C1CCOc2ccccc21)NC(N1CC(C(=O)OC)C(c2cn(C)cn2)C1)=O C1(OC)CC(CF)N(C(=O)CN(C(C2CC(O)C(F)C2)=O)CC2CC2)C1 c1(C(N(C)CC2N(C(CCC3CC(C)C3)=O)CCOC2)=O)c2c(nn1C)CCC2 N1(C(C2C(C)C2)=O)CCC(CNC(c2cc3sccc3n2C)=O)C(F)(F)CC1 c1(C(=O)Nc2cccc(C3CCCCC3)c2)cc2cc(Cl)c(Cl)cc2[nH]1 C1(C(N2CC(CCNC(C3N(CC)CC3)=O)(OC)C2)=O)CCC(F)CC1 c1(C(N2C(C(=O)NCC3(O)CCC(C)C3)C(O)CC2)=O)c[nH]c2ccncc12 Cc1ccc2ncc(C(=O)N(C)CCN(C(=O)CC(C)N3CCCC3=O)C)n2c1 c1(NC(C2CC3CC3N2C(c2cccc3c[nH]nc23)=O)=O)cc(F)c(F)cc1I N1(C(CC(CC(=O)Oc2ccc(OC)cc2)(C)C)=O)CC2CC23CCCC(C3)C1 C(C(O)CN=c1ccnc[nH]1)NC(=O)Cc1ccc2nc(O)[nH]c2c1 c1(C(N2CC3(CNC(=O)C(F)F)CCC2CC3)=O)ccccc1S(=O)C(F)(F)F C1(C(=O)NC)C2CN(C(=O)C(=O)Nc3ccccc3)CC12 N1(C(C(C)O)=O)CC2C(NC(c3cc(O)cs3)=O)C2C1 CC1CCc2ncc(C(N3CC4CC(NC(=O)COCCCF)C3C4)=O)n2C1 NS(=O)(=O)CCCCCCC(=O)NCC1(O)CN(C(C2CCCCC2)=O)C1 Cc1oc(C)c(S(N)(=O)=O)c1C(=O)NC1CC(C)(NC(c2nn[nH]c2Cl)=O)C1 C1(C(=O)NCC(=O)OCC#C)CCCN(C(=O)CC2CCCOCC2)CC1 S(=O)(=O)(c1ccc(=NCc2c(C)nn(C)c2C)[nH]c1)N(C(C(CC)CC)C)CC CCCCC(O)CC(=O)N(C(C)(C)CC(=O)NCc1ccnc(C)c1)C c1(N2CCCC(CCOC)(OC)C2)ccn2ncc(S(=O)(=O)N3CC=CC3)c2n1 C1(CC(=O)NCC(C2CCOC2)NC(c2ccncc2)=O)CCC2(CC2)CO1 N1(C(C)=O)CCOCC1C(=O)NC1CCCCC1NC(=O)CSC(F)(F)F CC(C)(C)C(CC(=O)NC1CCC2CC1CN2C(=O)C#CC1CC1)C(F)F CC1CCC=C1C(=O)NCC(O)CC1(C)CCCO1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCC1(NC(CCCC)=O)CC1 C1(c2n(CCSC)nnn2)(Nc2sc(Cl)nc2Cl)CCCN(C(C)(C)C)C1 C1(C)(C(N2CC(CC(CNC(COc3cc(C)on3)=O)(C)C)C2)=O)CCC(=O)NC1 c1(C(=O)NCC(C)(C2CC2)NC(C2CCCC2c2nc(S)n[nH]2)=O)csc(O)n1 c1(C(=O)NC(c2occ(C(N(C3CCC(C)C3)C)=O)n2)C)ccccc1O c1(C(N2C3CN(C(CCCC(=O)OC)=O)C(CC3)C2)=O)cnc2ccccc2c1 C(C1c2ccccc2CN1C)NC(N1CCCC(C(=O)NCCOC)C1)=O C12(C(=O)NC3CC4CC(OC)C4C3)CCCC1CN(C(c1cc(C)c(C)[nH]1)=O)C2 c1(C(C(=O)NC2CN(C(c3c(C)cno3)=O)CC2O)O)ccc(F)cc1F CC1CCC(NC(=O)CC2CCN(C)C2=O)CN1C(C1CSCN1C)=O C(=O)(C1=CC2(CCN(C(C3(F)CCCC3)=O)C2)C1)N1CCN(C(C)C)CC1 C(=O)(CCCC(=O)NCC1(NC(=O)COC2CCOC2)CCOC1)OC(C)C C(=O)(C(C)CS(C)(=O)=O)NC1CC2(C(NC(Cc3c(C)nc(C4CC4)s3)=O)C2)C1 C(C(CO)N=c1nc2[nH][nH]cc-2c(O)n1)NC(=O)CCF N(C1CCCOc2c1ccc1ccccc21)Cc1cc(Br)c(I)cc1 c1(CC(C)C)nc(C(=O)NC(CNC(=O)C(C)(O)C2CC2)CO)cs1 c1(C(=O)NC(CN(C(CN(C2CC2)CC)=O)C)C)n[nH]cc1F C1(C(=O)NCc2n(C)ncc2)CC12CCN(C(=O)COCC1CC1)C2 C1(NC(c2cccc(OC)n2)=O)CC12CCN(C(=O)CC(C)C(C)C)C2 CC1(C)CCC(C(N2CC(NC(c3ccc(CCF)cc3)=O)C2)=O)O1 Cc1cc2cc(NC(=O)Nc3nc(-c4ccc([N+](=O)[O-])cc4F)cs3)ccc2s1 N1(C(c2cnn(C(C)C)c2I)C(=O)NCc2cccs2)CCC(C)(C)C1C N1(C(c2cc(COC)sc2)=O)CC(OC)CC1CNC(c1ccnc(C)c1)=O Cc1cc2ncc(C(=O)NCC34CC(CO3)N(C(c3ccccn3)=O)C4)cc2[nH]1 C1(C(N2C(CN(C(=O)Cc3cnsc3)C)COCC2)=O)CC2CC1C1C2C1(F)F CCC(CC)(CO)C(=O)N1CC=CC(NC(=O)C=Cc2cscn2)C1 C=CCC(CC(C)C)C(=O)NCC1CC2CCC1N2C(=O)Cc1ccc(O)cn1 C(=O)(C=CS(C)(=O)=O)NCC(Cc1ccccc1)N(C(C(C(C)C)F)=O)C c1(CC)ncc(C(N2CCN(C(c3c[nH]c(Br)c3)=O)CC2)=O)c(O)n1 C(CN=c1cc(C2CC2)nc(Cl)[nH]1)NC(C(CCC)OCC)=O C(=O)(C1=CSCCO1)N1C(CCNC(c2ccn(CC#N)n2)=O)CCC1 C1(CC)CN(C(C2(COC)CN(C(=O)C3=COCCC3)C2)=O)CC12CC2 C(=O)(C(C)CC(F)(F)F)NC(C(C)C)CNC(c1ccc(CN(C)C)nc1)=O Cc1cc(F)c(C(=O)N(CC(C)CNC(C2CC3CCC2O3)=O)C)c(Br)c1 c1(C(=O)NCC(=O)NCC2CC2)ccc(CNC(C2CC(O)C2)=O)s1 Cc1cc(C(N2CC(NC(c3cc(C)n(C(F)F)n3)=O)C(O)C2)=O)c(N)cc1F c1(-c2ncsc2)cc2c(s1)CCN(C(=O)NCC)C2.C(C(C)NC=O)OCC C1(NC(c2c(CC)noc2)=O)CCN(C(=O)Cc2ncc(Cl)s2)C1C c1(CNC(CS(CC)(=O)=O)C)ccc2c(c1)SCC(=O)N2 C(=O)(C(C)(C)Cc1cccc(Cl)c1)NC(C)CNC(C1CNC(=O)N1)=O c1(SC)ncc(C(=O)NC(CO)C(C)NC(C2C(C)(C)C2(F)F)=O)c(O)n1 C(c1cnccn1)=CC(=O)NCC(CNC(c1ncnn1C(C)C)=O)OC c1(C(N2CC(NC(C3CSC3)=O)(CO)C2)=O)ccc(Cl)cc1Br N(C1CCc2cc(CNC(c3ncsc3C(F)(F)F)=O)ccc21)C(C1C(C)C1)=O Cc1c(F)ccc(CN2CCC(O)(CC(=O)Nc3nc(Cl)nc(Cl)n3)CC2)c1Cl N1(C(C2CC(OC)CN2C(c2ccsc2)=O)=O)CCC(O)C12CCC2 c1(NC(C(=O)NCc2nnc3n2CCC3)=O)cc2ccccc2s1 N1(C(c2c(C)con2)=O)CCCCC(CNC(=O)CCC2CCCCO2)C1 c1(NC(=O)NCC(CN(C)CCO)O)c(OC(C)(C)C)cc(Br)cc1F C(N=c1nc(O)c2ccccc2[nH]1)C1CCCN(C(C2(C)CCCCO2)=O)C1 C12(CN(C(C3CC(CC)(CC)C3)=O)C)CC1CN(C(c1ccnn1C(F)F)=O)C2 N1(C(CC2CCC(NC(C3CC34CCCCC4)=O)CC2)=O)CC2(CCC2O)C1 N12CC(NC(=O)C(COC(C)C)NC(C)=O)CC1C2.CCC(C)=CC(=O)OCC CC1(C)OCCNC1C(=O)Nc1ncc(Cl)cc1F Oc1c(F)cc(CNC2(c3nnnn3CC3CC3)CC(F)(F)C2)cc1F c1(NC2CCN(CCOC)C2)ncnc2[nH]c3cc(F)ccc3c12 C1(C(N2C(CN(C(c3c(CC)onc3)=O)CC)CCCC2)=O)CCN(C)C(=O)C1 c1(OC)ccc(CN2CCC2C(=O)Nc2cnn(C3CCCC3)c2C)cc1Br C1(CC)CC(C(=O)N(C)CC2CC(O)C2)CCN1C(c1cc(C)cs1)=O C1(CC(=O)NC(C(CO)SC)C)(NC(=O)CN2CC3CCC2C3)CCCCC1 Cn1nc(C(N2CCCC(CO)(NC(=O)C(C3CCOCC3)F)C2)=O)cc1C#N N1(C(c2c(CC)non2)=O)CC(C)(C)CC1C(=O)NCCNS(=O)(=O)CC c1(OC)c(C(=O)C(c2cnn(C)n2)C#N)c(CNC(=O)OC(C)(C)C)nn1C CCC(F)(F)C(C)(C)C(=O)NCC1(C)CCC(NC(c2cnc(SC)s2)=O)C1 C(=O)(C1=CC2CCC(C1)C2)N1CC(CC(C)NC(=O)CN2CC3CC3C2)C1 C(=O)(CC1CCc2ccccc21)C(CNC(=O)OC)=O.C1(NC)CCN(CC)C1 C(C(CNC(c1cc(C2CCC2)[nH]n1)=O)S(C)(=O)=O)NC(CCCOCCC)=O Cc1nc(C(=O)NC2CCCC(NC(C3(CO)CCC3)=O)C2)ccc1Br C(C1CC(=O)Nc2ccccc21)NC(C(C)NC(c1ccc(Cl)c(Cl)c1)=O)=O c1(OC)ncc(C)cc1NC(C1CC=CC(NC(C2CNC(=O)O2)=O)C1)=O c1(C(=O)NC2CN(C(C(CC)F)=O)CC(C)(C)C2)cc2c(Cl)cncc2s1 c1(CC(=O)NCC(=C)Br)ccc(-n2cc(COC3CCOC3)nn2)cc1 CC(C)CC(C(=O)N(C)CCNC(=O)C(C)C(F)(F)C(F)F)C(N)=O CC12COCC1(C)CN(C(=O)CCC1CCC(NC(c3c[nH]c(=N)o3)=O)C1)C2 N1(C(=O)CCn2cc(COc3cccnc3)nn2)CCC(O)(C(Cl)(Cl)Cl)C1 C1(C(=O)NC(CC=C)C2CC2)CC(O)C(O)CC1CNC(=O)CC(C)C(=O)OC N1(C(C2C(C=CC)CN(C(=O)CCCCCOC)C2)=O)CC2CCC1C(O)C2O CCCCC(CNC(=NCCOC)NCC(C(F)F)c1ccccc1)CC c1(N2CC(C)(NC(CCCCC(C)C)=O)C2)nc(Cl)nc2cccc([N+](=O)[O-])c12 C1(CN(C)C(c2sccc2C2CC2)=O)C2CN(C(c3csc(=N)[nH]3)=O)CC12 C1(OC)CC(CN(C(=O)CC2CCC(=O)C2)CC)N(C(=O)CN(C(=O)C(C)C)C)C1 N1(C(C(C(CC)C)O)=O)CCC2(CC1)CC2NC(c1ccsc1)=O C(=O)(C(CNC(C1CCOC(C)(C)C1)=O)C(C)(C)C)N(CCN1CC=CC1)CC c1(C(N2C(CNC(CCCC(=C)C)=O)C(O)C(O)C2)=O)cc(S(N)(=O)=O)oc1C N1(C(C(N2CCC(C)C2)=O)=O)CC2OCCN(C(=O)CCc3nncs3)C2C1 N1(C(CC(CC)(F)F)=O)CCOC2CN(C(C3CCC34CCC4)=O)CC12 n1(CC)nc(C(=O)N(C)CC2COCCN2C(=O)C=CSC)cc1C1CC1 C1(CC)CN(C(C2(OC)CCOCC2)=O)CCN1C(c1csc(Cl)n1)=O C(N=c1cc(C#N)[nH]c2ccccc12)c1ccc(OCC=C)cc1 N1(CC(=O)NC2CCC2NC(c2ccc(=O)oc2)=O)C(=O)CCCC1=O C1(CNC(CSCC#C)=O)(OC)CCN(C(=O)CC2CCOC2(C)C)CC1 N1(C(C2(SC)CC2)=O)CC(CNC(=O)C(C)Oc2ccc(C#N)cc2)C2(CC2)C1 CCCCC(C)C(=O)N1CC(NC(c2cc(N)cnc2C)=O)C(C)C1 c1(C(=O)NC2CN(C(C3(C=C)CC3)=O)CC2O)cccc2c1oc1ccccc21 N1(C(Cc2n(C)nnc2)=O)CC=C(C(=O)NC2C=CCC2)CC1 c1(C(N2CC(O)(CCNC(C(CO)OC)=O)C2)=O)cnn(C(C)C)c1C CCS(=O)(=O)C=CC(=O)NC1CCC(CNC(c2cc(CO)[nH]n2)=O)C1 c1(CC)nc(=NCCC2CCC(NC(=O)Cc3c(C)nn(CC)c3Cl)C2)s[nH]1 C(c1ccc2c(c1)COCC2)=Cc1onc(CC)n1 Cc1ccsc1C=CC(=O)NC(C1CCCC1)CNC(=O)C(C)CF c1(C(C(=O)NCC2CCN2C(=O)C(C)C2CC2)OCC)ccccc1 N1(C(C(CCC)C)C(=O)NCCC2CC2)CCc2cc(C)cc(C)c2C1 C1(CC)C(C(=O)NC(c2ccnn2C)C)CCN1C(=O)C(CCOC)OC N1(C(c2n(C(C)C)ncc2)=O)CC(C2(NC(C3CCCSC3C)=O)CC2)C1 N1(C(C(CC)F)=O)CC2CCC1CN2C(c1c(C)nn(C)c1-n1ccnc1C)=O C1(C(=O)NC2COC(C(C)C)C2)(NC(CC=C)=O)CCN(C)C1 C(=O)(CCN=C(NCc1nccs1)NC1CC1(c1ccccc1OC)C)NC N1(C(CCc2cc(C)on2)=O)CCC(F)(CNC(C2C3COCC23)=O)CC1 C1(NC(=O)Cc2ccc(C(F)(F)F)cc2F)CC2CN(C(=O)CSC(F)F)CC2C1 Cc1cc(C(N2CC(CCCCNC(=O)CCCC3CCC3)C2)=O)c(N)c(F)c1 Nc1cc(C(=O)NCC2CN(C(c3ncc(Cl)s3)=O)C2)nc(O)c1 C1(NC(c2c(CC)nco2)=O)CC2CC(C1)N(C(=O)CC1CC(C)(C)C1)C2 C1(NC(C(=Cc2cnc[nH]2)C)=O)CC2CCC(C1C)N2C(c1cccn1C)=O N1(C(C=CC)=O)CCn2nc(C)c(CNC(=O)COc3cccnc3)c2C1 CC1(C)NC(=O)CC1C(=O)NCCC1(NC(c2cc(C(N)=O)[nH]n2)=O)CCCC1 c1(OC(C)C)cccc(NC(C2COCCC2NC(c2cc[nH]c2)=O)=O)c1 c1(-c2n(-c3cccc(SC)c3)nc(C)n2)cc([N+](=O)[O-])cnc1O N1(C(CC2C(C)CC2)=O)CCC(C2(O)CN(C(=O)C=CCn3cncn3)C2)CC1 N1(C(CC2(NC(=O)Cc3cnns3)CC2)=O)CC2CCC=CC12 CC1C(NC(c2cnc(C3CC3)[nH]2)=O)CCCN1C(c1cn2ccnc2s1)=O C1(F)(C(=O)NC2CCN(C(N(C)C)=O)CC2)CNCC12CCC2 N1(C(C2CCN(C)CC2)C)CCCC(O)(c2cn(C3CCC(O)CC3)nn2)CC1 c1(C(N2C3C(NC(C(C=C)(C)C)=O)CC(C3)C2)=O)cc(C)cc2ccncc12 C12(CCCC1)c1cn(nn1)C(C)C(=O)N2.C1(C(=O)NCCOC)CCCCC1 CCCCC(CNC(C1CCCCN1C)=O)NC(=O)CC1CCCC1C N1(C(C(CCC)C)=O)CC(NC(c2ccccc2OC2CC2)=O)CC2(CCC2)C1 Cc1cc(C(N2CCC3CC2CN(C(C2(C)CCCO2)=O)C3)=O)cc2nc[nH]c12 CC(C)CC(C(=O)N1CC=CCC1)ONC(c1cccc(F)c1F)=O C1(NC(CC2(CC)CCOCC2)=O)CN(C(c2cccnc2O)=O)CCC1C Cc1cc(C(=O)NCC(CC(C)C)NC(C2CC3(C2)CC3F)=O)oc1C C(=O)(C(C)(C)C(c1ccccc1)OC(=O)C(O)Cc1ccccc1Cl)OC(C)C CC1(C)CCN(C(C2CCC(=O)C2)=O)CC1CNC(c1coc(Br)c1)=O c1(SC)cc(C(=O)NC2(CO)CN(C(c3coc(C)n3)=O)C2)ccc1NC(C)=O N12CCc3ccc(cc3C1)O2.Cc1cnccc1CNC(=O)Nc1ccccc1 c1(C(=O)NC2(CC=C)CCN(c3ncns3)CC2)cc(C)nc2onc(C)c12 N1(C(CC)=O)CC(F)(F)CC1(C)CNC(=O)Cc1ccc2nc[nH]c2c1 N1(C(CCCC=C)=O)CCC(C)C(CC(=O)N(CCC)C(C)C)C1 C1(NC(C2C(C)(C)C2)=O)CCC(F)(CNC(=O)CC2(N3CCCC3)COC2)C1 C1(CNC(C2CS(=O)(=O)C2)=O)CCN(C(c2cnn(CC3CCOCC3)c2)=O)C1 C1(C(=O)NCC2(CCNC(C3C(CC)C3C)=O)CC2)CC(=O)N(C(C)C)C1 C1(NC(CCOCC)=O)CC2CCC1(C(=O)N(CC(=O)OC)C1CC1)C2 CN=c1[nH]c(C(=O)NC2(CCNC(c3cncc(OC)n3)=O)CC2)cs1 c1(CCOCC)nc(C(N2CCC(CN(C)C(C3CC3COC)=O)C2)=O)co1 Cc1csc2cc(C(N3CCC(C(C)NC(=O)CC(C)P(C)(C)=O)CC3)=O)[nH]c12 CC1CCN(C(=O)C(C)(C)C#N)CC1NC(=O)CC1CCCCC1 c1(C(N(C(CNC(C2(C)CC(=C)C2)=O)C)C)=O)ncc(C)cc1F C1(CC(=O)NC2(CC(=O)OC)CC2)C2CCCC2N1C(c1cccc(C#N)c1)=O c1(CC)scnc1C.C12CC(C1)CC(=O)NC(C1CC1)CN2C(=O)CN1CCCC1 C1(C(=O)NCCC(C)NC(COCC)=O)CCCC(=O)CC1 N1(C(CCc2c(C)noc2)=O)CCC(C)C(N(C(=O)CCc2ccncc2)C)C1 Cc1ccc(Cl)cc1OCC(=O)NC1CCC(C)N(C(=O)CC2CC(F)C2)C1 n1(CC(=O)N(CCC(=O)NCCCc2cnc[nH]2)CCO)ncccc1=O Cc1nn(CC(=O)NCC(CNC(C2(CC(C)C)CCC2)=O)CO)cc1Cl CCCCCC(=O)NCC(=O)NCC1COCCN1C(c1ccc(CSC)o1)=O N1(C(c2c(C)occ2)=O)CC(CNC(C2(n3cccn3)CCCC2)=O)C(F)(F)C1 C=CC1CN(C(c2c[nH]nc2CNC(C2CCCC(OC)C2)=O)=O)CC1O C1(NC(C2C=CCCC2)=O)C2CCC1N(C(=O)Cc1ccsc1)C2 C(=O)(CC(CC)c1ccccc1)NCC(CNC(c1c(CC)cco1)=O)OC S(=O)(=O)(c1ccccc1F)N1C(CNC(=O)Cc2c[nH]c3cccnc23)CCC1 Cc1c(C(=O)NC2CCCC2NC(=O)CCCC2CCC2)[nH]c2c1C(=O)CCC2 N(C(=NCCC(C)C)N1CCC(c2ccccc2F)C1)CCC(C)=O N(C1CCc2cc(Cl)ccc21)C(c1c(Cl)cncc1Cl)c1n(C(C)(C)C)nnn1 N1(C(CC2(CNC(C(C)NC=O)=O)CC2)=O)CC2CC=CCC2C1 c1(CC(=O)NC(C)CN(C(=O)CCC2CCCC2)C2CC2)ccc2oc(O)nc2c1 C(=O)(C1=CCC(NC(=O)C(c2ccccc2)O)C1)N1C(C)(CCO)CC1 C1(NC(c2ccc(Br)cc2)=O)CN(C(C2(CF)CC2)=O)CC1n1cccn1 c1(C(=O)OCC)cc(C)nnc1N(CC(C)NC(=O)C(C)C(C)CC)C N1(C(C2C(C=C)C2)=O)CCC2(CCCC2CNC(=O)CS(N)(=O)=O)CC1 S(=O)(=O)(c1ccc(N2CCc3sc(C)cc3C2)cc1Br)N(C(CCC)C)C C1(C(N(C)C)=O)CCN(C(=O)NCC2C=CCCC2)C1 N1(C(CC(=C)C)=O)CCCC12CCN(C(C1CC(=O)N(c3cn[nH]c3)C1)=O)C2 N1(C(C(F)=C(C)C)=O)CCN(CC2(NC(C3COC(=O)N3)=O)CC2)CC1 c1(C(=O)NC(C(=O)N(CC(C)NC(=O)C2CC2)C)C)ccc(S(=O)(=O)NC2CC2)o1 c1(C(=O)NCC(COC)OC2(CO)CC3CCC2C3)c(C)ncnc1C N1(CC(N2C(CN(C)CCc3cccc(F)c3)CCC2)=O)C(=O)CNC1=O CC1CN(C(=O)CCn2cccn2)CCN1C(=O)CC1CC=CCN1C C1(N(C(C2OCCC2C)=O)CC)CCN(C(c2ncsc2Br)=O)C1 c1(C(N2CCCN(C(c3cc(C)sc3C)=O)CC2)=O)cnn2c1CC(F)(F)C2 C(=O)(C1=CCOCC1)N1CCC(C(N2CCC(C)(NC(C)=O)C2)=O)C1C(C)C S(=O)(=O)(c1ccc(NCC(C)F)c(F)c1)NCCCN(CCC)CCC Cc1cc(C(=O)NCC2CC3CN(C(c4cnc(C)o4)=O)CC23)c(O)nc1C c1(C2(C(=O)NC(CNC(=O)CC3(O)CCOC3)CO)CCC2)ccc(F)cc1 NC(=O)CC(O)C(=O)C(N)=O.N1(C(c2scc(CN)c2)=O)CCCC(N=O)C1 c1(NC(=O)Nc2cccc(C3OCCO3)c2)ccc(C2CC2)nc1 C12(C(=O)NC3(C)CC3)CC(CO)(C1)OC2(C)C.N12CCC(C1)N(CCO)CC2=O c1(C(N(C(C)CNC(=O)Cc2nnc(S)n2C)CC)=O)cc(OC)n(C)n1 Cc1sc2ncnc(C(=O)NC3(C)CCC(NC(=O)CCC(C)C)CC3)c2c1C N1(C(Cc2ccc(C(C)=O)s2)=O)CC2OCCCC2(C=O)C1.C(C)(C)(C)O N1(C(c2c(C)cc(CC)o2)=O)CC2CCCC1CN(C(c1cc(Cl)nn1C)=O)C2 C(CNC(=O)COOCO)(CC(F)(F)F)NC(C1(OC)CCSC1)=O.c1ccccc1 C(=O)(CCCCC(C)(C)C)NC1CC(CNC(C(C=C=C)C)=O)CC1O c1(C(=O)NC2CN(C(C3CCCS3)=O)CC2F)ccc2nccnc2c1 N1(C(c2c(C)oc(Br)c2)=O)CCN(C(=O)CC2C(C)(C)C2(C)C)C(C)C1C CC(C(=O)NC1CC(CCNC(=O)Cn2cc(C3CC3)nn2)C1)C(C)(C)C c1(CN(C(c2csc(-c3cccs3)n2)=O)Cc2nn[nH]n2)nc2ccccc2[nH]1 c1(OC)ccc(CC(C)C(=O)NC(C)(C)CCNC(c2cncs2)=O)cc1 C(=O)(C1CCCc2cncn21)NCc1c(CN(C(C2(OC)CC2)=O)C)cccc1 c1(C(=O)NCC2(F)CN(C(c3cc(C)c(F)cn3)=O)C2)nn(C)c(=O)cc1C C1(C(C)NCCCN2CCCC(O)C2)CCc2nnc(C(F)F)n2C1 C1(CCOC)(NC(=O)C=CCO)CCN(C(=O)C(O)CC2CCCCC2)C1 N1(C(Cc2c(C)nc[nH]2)=O)CC2(CCC2)CC1CNC(c1cc(Br)co1)=O C#CCC(C(=O)N1CCCC1(C)CCCO)NC(C1CS(=O)C1)=O C1(C(=O)NCCC2CC(NC(C3CC4CC4C3)=O)C2)CC2COCC(C1)C2(F)F c1(CC(N2C(C(=O)NC3CC(CC)(CC)C3)CC2)=O)ccc(Br)cc1 c1(CNC(C=C(CC)CC)=O)ccnc(OC)c1.C12(CSC1)C(=O)N2 Cn1cc(Br)c2c(C(N3CC(C)(C)CC3CNC(=O)CCF)=O)ncnc12 N1(C(=O)OCCC(C)C)CC2CN(C(=O)CCCc3ccc(Cl)cc3)C2C1 C(C(C)(CC(C)C)NC(=O)C(=CC1CCCC1)C)NC(C(C)OCCOCC)=O N1(C(c2cccc(SC)c2)=O)CCC(NC(c2ncsc2C2CC2)=O)C(F)C1 N1(C(c2cc(O)ccc2O)=O)CCC(F)(F)C(Nc2ncccn2)C1 C(=O)(CC(C(F)(F)F)n1ccnc1)NCC1(O)CN(C(=O)OC)C1 CC1=C(C(=O)N2CCN(C(=O)C(C)C#N)CC2C2CCCC2)CCC1 CCCCC(C(=O)N=c1cc2ccccn2[nH]1)NC(=O)C(O)C(F)(F)F N1(C(C(C)OC)=O)CC(CNC(=O)Cc2ccn(CC(C)C)n2)CC1(C)C c1(CCC(=O)NC(C2CCCN(C(=O)C(C)(C)C#N)C2)C)c[nH]c2ccccc12 N1(CC(C)C)CCCC(C(N2CCCCC2CN(C(=O)CC(C)(C)C)C)=O)C1 c1(NCC2CN(C(c3cc(CCOC)on3)=O)CC2C)ncnc2c1CCC2 CCS(=O)CC(=O)NC(Cc1ccccc1)CCNC(c1cnc(C(C)O)s1)=O c1(C(N2CC(NC(C(c3ccccc3)C)=O)C(O)C2)=O)cc(Cl)c(F)cc1F C(=O)(CCOCCNC(=O)Cc1ccon1)NCC(=C)F c1(CN2CC(C)N(C(C34CCC(CC3)CC4)=O)CC2)ccc2c(c1)OCO2 c1(C(=O)NCCC(CCNC(C(=Cc2cnc[nH]2)C)=O)C)cc(CO)ccc1Cl c1(N(CC(=O)N(CC)CC)C=O)c(F)c(F)c(Br)c(F)c1F C1(CNC(=O)C=Cc2cnc[nH]2)CCCN(C(C2CCCCC2)=O)C1 c1(C(N2CC(CCNC(c3c(C)snn3)=O)OC(C)C2)=O)ncnc2c1CCC2 C1(CNC(C(C2CN(C(C)=O)C2)O)=O)CCNC1=O C1(F)(C(=O)Nc2cc(CC3CC3)on2)CCC(CNC(=O)CSC2CC2)CC1 C1(CC)CC(CC(N2CC(CNC(=O)C(C)CCc3ccccc3F)C2)=O)CCO1 C=Cn1nccc1C(=O)NCC1CCC(NC(c2sccc2OC)=O)C1 C1(c2n(CC)nnn2)(NCC(c2ccccc2OC)OC)CCC(C)SC1 C(=O)(CCC(CF)CF)NC(C(=O)NC(c1ccn(C)n1)CC)CCN(C)C C(=O)(C(C)(C)CC(F)F)N(CCC1CCN(C(C2(C)CCC(C)C2)=O)CC1)C C1(C(=O)NCC(C)NC(C2C(C)(CC)C2)=O)CSCCS1 C1(C(C)C)CN(C(c2scnc2Cl)=O)CCN1C(C1CCCN1C)=O c1(C(=O)NCC2C(CC)CCN2C(=O)Cc2cnn(C)c2C)nnc(O)nc1O c1(C(N2C(CNC(COCCOCC#C)=O)CCC2)=O)cnc2c(ccn2C)c1 c1(C(=O)NC2CN(c3ncncc3Br)CCC2(F)F)cccc2nc(Cl)sc12 C(C(C(=O)NC(C)C(=O)NC1CC1)C(C)C)NC(c1cc(CC)no1)=O C12(C(=O)OCc3cc(C)on3)CCCN(C(=O)OC(C)(C)C)C1C2 C1(CC(=O)NC2CN(C)C(CO)C2)C2CCCC2N1C(c1cnn(CCO)c1)=O c1(C(=O)NC)cccc(CNC(c2ccc(CCC)cc2)=O)c1C CC1COCC2(CCC2)N(C(=O)Cc2cc(C(F)(F)F)cc(Cl)n2)C1 N1(C(c2ccc(C)o2)=O)CCCC2(CCCN(C(c3cc(Br)ccc3Cl)=O)C2)C1 C(=O)(C#CC1CCCCC1)N1CCC(N(C(c2cc(CC)ncc2)=O)C)C1 c1(C(=O)NC2CCC(NC(CC3C(C)(C)CCO3)=O)CC2)cccc2ncsc12 CCC(C)C(C(=O)NC1CC(CNC(=O)COCC(F)F)C1)c1ccccc1 CC(CC(=O)NCCn1cc(C(=O)NCC2CN(C(N)=O)C2)nn1)C(F)(F)F N1(C(C(CC#C)NC(=O)C(C)OC)=O)CCC(c2ccccc2)(CN)CC1 C12(C(=O)NCC(CC)(CC)NC(c3csc4nnsc34)=O)CCCCN1CCC2 CC(CCC(C)(C)C)C(=O)Nc1ccccc1-n1cc(CN(C)CC2CC2)nn1 C(=O)(C(C(=O)NCCCC(C)NC(=O)CN(C)C(c1ccsc1)=O)OC)OC c1(C(=O)NCc2ccnc(-c3nn[nH]n3)c2)ccc(Cl)c(C2CC2)c1 c1(NC)ccc(Cl)c(C(=O)NC2CN(C(C3CCCCC3C)=O)C2)c1 N1(C(C2CCC(C)(C)C2)C(=O)NC(c2ccccc2)C)CCC12CCSCC2 c1(CC)cn2c(C(=O)NCC#CCNC(=O)CC3(O)CCCCC3)cccc2n1 O=C(N=c1[nH]nc(Cl)cc1O)c1occc1OC(F)F C1(NC(c2ccc(OC)o2)=O)C=CCN(C(=O)Cc2ccc(C(C)=O)s2)C1 C1(C(N(C(C)CN(C(=O)C(C)Cn2cccn2)C)C)=O)CC(S(C)(=O)=O)C1 N1(C(C)=O)CCCCC1C(N1CCCCC1CCNC(=O)CCn1ccnc1)=O CC(CNC(=O)CCCF)(CO)NC(=O)CCCc1ccsc1 CC1Cc2cc(CC(=O)NCC(C)(C)CNC(C3CCS(=O)(=O)C3)=O)ccc2O1 Cc1ccc(OCCC(=O)NC(C)(CNC(=O)CC2CCCCO2)C(C)C)cc1 Cc1cc(C)c(C(=O)NCC2(C)CCN(C(C3CCCOC3C)=O)CC2)c(O)c1 C1(CC)(NC(c2coc(O)n2)=O)CCN(C(c2ccc(C)nc2C2CC2)=O)CC1 C(=O)(C(C#N)C(C)(C)C)NC(CC)(CNC(=O)COc1ccc(F)cc1F)CC c1(C(C)C)cccc(NNC(=O)Nc2ccc(C3CC3)c(F)c2)c1 c1(C(Cn2c(N3CCCC(NC(=O)OCC)C3)nnn2)(C)O)cc(Cl)ccc1Cl Cc1cccc(C=CC(=O)NC(CNC(=O)C(N2CCSCC2)C)C(C)C)c1 C1(N(C(C)(C)C)C(=O)CC2CCOC2)CCN(C(=O)NC2(C)CCCS2)CC1 N1(Cc2cccs2)CC(C(=O)OCC(C)OCC)CC1=O N1(C(C(CC)C#N)=O)CCCC2CN(C(c3cn(CC4CC(=O)C4)nn3)=O)CC12 N1(C(C(F)=C(C)C)=O)C(C(=O)NCc2nc(O)ccc2C)CC2CCCC12 C1(C(C)OC)CCN(C(C2CCC=CC2NC(C2CCCN(C)C2)=O)=O)CC1 O=C(O)C(F)(F)C(c1ccccc1)NC(C1CCCCO1)=O c1(CC(N2CCN(C(c3noc(CC)c3C)=O)CC2)=O)ccc2ncsc2c1 N1(C(c2c(CC)cnn2C)C(=O)NCCOCC)CCC23CCC(CC12)C3(C)C c1(C(=O)NC2CC2CNC(C(CC)C(C)O)=O)ccc2oc(C)nc2c1 C=CC1(C(N2CCN(C(C3CC3F)=O)C(c3cn[nH]c3)C2)=O)CCCCC1 C(CC(=O)NCC1CC2C(C1)C2(F)F)(C(C)(C)C)NC(C(C(C)(C)C)=O)=O c1(OC)ccnc(OC)c1C(=O)NCC(O)CNC(c1cc(F)cs1)=O C1(NC(c2cnc(C(C)(C)C)o2)=O)CCN(C(=O)CCc2cnn[nH]2)C12CC2 c1(C(N(C)C)=O)cccc(OC(F)F)c1Cl.n1(CCCO)cc(C2CC2)nn1 C1(NC(C(=O)Nc2cc(Cl)c(Br)cc2F)=O)CCc2nnc(O)cc2C1 C1(C(N2CC(C)(NC(c3cccc(CC)c3C)=O)C2)=O)CCc2cnnn2C1 c1(C(N2CCN(C(c3csc(C)c3N)=O)C3C2C3)=O)ccc(S(N)(=O)=O)o1 C1(NC(C2(CCC=C)CC2)=O)CCN(C(=O)CN2CC(C)(OC)C2)C12CC2 Cc1cc(C)c2nc(NC(=O)CNC3(C4CNC4)CCC3)sc2c1 N(C(=NCc1ccccc1)N1CCCC(O)CC1)C(C1(Cl)CCOCC1)C C1(CC(=O)NC(C)C(CO)NC(C2CN(C3CCOCC3)C2)=O)CCCOCC1 c1(NC(C(N2CCC(CO)C(O)C2)c2n(C)nnc2)=O)cccc([N+](=O)[O-])c1 Cc1nc(C(=O)NC2CCN(C(C3CCCN(C(=O)C(C)(C)C)C3)=O)C2)nn1C CCC(CN(C)C)C(=O)NC1CCC1NC(c1cccc(O)n1)=O C1(NC(C(=O)NCC)=O)CC2CC1CN2C(C1CCCN1C(C)C)=O c1(OC)nc(C)ccc1C(=O)N(CCCCCNC(C1CC(C)N(C)C1)=O)C N1(C(C2(F)CCN(C(c3c(C(C)C)occ3)=O)C2)=O)CCOC(C)(C)C1C CC(CCC(C)(C)C)C(=O)NC(C)(CO)C(=O)Nc1cccc(C#N)c1 C(C)(C)(C#Cc1cn(C2COCC2O)nn1)NC(C(C)c1ccco1)=O C1(C)(CNC(C2(OC(C)C)CCC2)=O)CCN(C(C2(C)CC2(F)F)=O)C1 CCC(C)(CNC(C1CCOC1=O)=O)NC(c1cc(C)c[nH]1)=O Nc1cccc(CCC(=O)NCC2CCCN2C(=O)Cn2cccnc2=O)c1 c1(CC(=O)NCCCCNC(Cc2cccc(SC)c2)=O)cccc2c1OCO2 N1(C(c2ccccc2F)=O)CCOC(CNC(C2(CO)CCC2)=O)C1 c1(C(N2CCC(O)(CNC(C=Cc3scc(C)n3)=O)C2)=O)cccc2oncc12 CC1CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CCC1CNC(c1ccc(=O)n(C)c1)=O CCCCCC(CC)C(=O)NC1(C(=O)N(CC(O)COC)C)CC(F)(F)C1 Cc1cc(C)n(-c2cccc(CNC(=O)NC3CC(F)(c4ccccc4)C3)c2)n1 CCCCCC(F)C(=O)NCC1(OC)CN(C(=O)C(C(C)CC)N(C)C)C1 Cc1cc(CCC(=O)NCCOC2CN(C(=O)C(F)CC3CC3)C2)cc(C)n1 N1(C(COC(C)=O)=O)CCCC12CCN(C(c1sc(C(F)(F)F)cc1C)=O)C2 c1(C(N(CCCN(C(=O)CC2CS(=O)(=O)C2)C)C)=O)ccc2nc(O)[nH]c2c1 CCC(CC(F)(F)F)C(=O)N1CCN(c2ccc(F)cc2C)CC1 C1(NC(C(c2scc(CC)n2)(F)F)=O)CN(C(=O)CN2C(=O)CCC2=O)CC1C C1(C(N2CC(C)(NC(=O)CCc3ccc(Cl)s3)C2)=O)(NC(C)=O)CCCC1 C1(C(N(C)CCOCCNC(C2CCCN2C)=O)=O)CS(=O)(=O)CCO1 C(=O)(CCCC(=O)C1CC1)N(CCC(C(C)C)NC(=O)CCCCNC(N)=O)C c1(NCC2OCC(CNC(c3c(CC)cno3)=O)C2)c(Cl)cccc1[N+](=O)[O-] C1(CC(=O)N(CC(C)(C)CO)C)CN(C(=O)CC2CCCC3CC23)CCO1 C1(C(=O)NCC2(COC)CCCC2)CCN(C(=O)C2(C#N)CCCOC2)O1 N1(C(c2ccnc(C)n2)=O)CCC(C)C(CNC(=O)C2=CCSC2)C1 Cc1ccc(-c2nc(C(=O)NC(C)CN(C(=O)Cc3ccsc3C)C)cs2)cn1 C1(NC(C2C(C)(C)C2)=O)CN(C(=O)CC2CCN(S(C)(=O)=O)CC2)CC1O c1(C(C)(F)C(=O)NCCCNC(=O)Cc2coc(C(F)F)n2)ccc(F)cc1 C(=O)(C1=CCCOCC1)N1CC2CC(C(=O)Nc3c(C)ccc(Cl)c3)(C1)C2 c1(C(=O)NCC2(CN(C(C(C(C)OC)O)=O)C)CC2)c[nH]c2cc(F)ccc12 CC1CC2CN(C(C3CC=CCO3)=O)CC2N1C(c1cnc2cccnc2c1)=O CCC(C(=O)N(C)CC1CC1Cl)C(C)C.C12(CC1)C(=O)N2 c1(C(N(CC(O)CNC(c2cnncc2O)=O)C)=O)cc2cccc(Cl)c2[nH]1 c1(OC)c(C(N2CC3CC2C3CNC(=O)C(C)C2CCCC2)=O)ccnc1Cl Cc1cccc2cc(NC(C3CN(c4nccc(C(N)=O)c4[N+](=O)[O-])C3)=O)[nH]c12 N1(CCc2cn(C(C3CC3(Cl)Cl)CC)nn2)CCC(Cn2nc(C)cc2C)CC1 c1(SC(C)C(=O)N(C2CC(NC(C3CC(O)C3)=O)C2)C)ccc(F)cc1 c1(C(=O)NCc2ccc(C)s2)cc(CNC(=O)CC2(C#N)CC2)ccn1 CC1CCN(C(C2C3CC(=O)CC23)=O)C1CNC(=O)C(C)(Cl)Cl C#Cc1ccc(C(=O)NCCCC(CC)CC)cn1 C(=O)(C(C)(C)C(=O)NCCN1CCN(C(C2CNC(=O)N2C)=O)CC1)OCC c1(C(N(c2ccc(CC)cc2)C)=O)ccc2cnn(C)c2c1 N1(C(c2csc(C(=O)OC)n2)=O)CC(OCC)CC(F)(F)C1 c1(C(=O)Nc2c(C)cccc2)cn2ccc(-c3ccnc(OC(C)C)c3)cc2n1 C1(NC(C(COc2c(OC)cc(C)cc2)(C)C)=O)CCN(C)C2(CC2)C1 C(=O)(CCC(C)(C)C)NCC1OCCN(C(c2cnn(C)c2Cl)=O)C1 C(=O)(C1=CCC(NC(=O)CC2C=CCCC2)C1)NC1(C(=O)OC)CCCC1 C(CC(=O)NCC1(C)CC2CC2C1)(C(F)F)NC(c1c(CC)c[nH]c1)=O CC(O)C(C)C(=O)N(CCCOCCNC(c1cc(C2CCCC2)nn1C)=O)C c1(OC)ccccc1C1(C(=O)NC(C)(C)CCNC(c2ccsc2)=O)CC1 S(=O)(=O)(c1ccnc(NC(=O)Cc2coc(-c3cccs3)n2)c1)N(C)C c1(CN2C(CC(=O)OC)CCC2)cc(F)ccc1NS(=O)(=O)CCBr C1(C(=O)NCCCCCNC(=O)CC2CCC=CCC2)CCN2CCCC2C1 CN1CCC(C(=O)NCC(c2ccccc2)CNC(=O)CC(F)F)CC1 C1(NC(=O)C=Cc2ccoc2)CC2CC1CN2C(c1cnsc1)=O CC1COC(C(N2CC(N(C)C(c3cc(C4CC4)on3)=O)C2)=O)C1 C1(F)(C(N2CCC(NC(c3nnc(C(C)(C)C)s3)=O)C2)=O)C2CCCC12 C=C1CC(C(=O)NC2(F)CCC2)(CNC(=O)NOCC(F)F)C1 c1(CC(=O)NC2C(NC(C(CC)SC)=O)COCC2)cc2ccccc2nc1O C12(NC(CCOCC#C)=O)CCC(CN(C(=O)CC(C)CC(=O)OC)C1)C2 c1(CCC(=O)NC(CC)CN(C(=O)C(C)Cc2ccncc2)C)nc(C)c(C)o1 C1(N(C(=O)Cc2ccoc2)CC)CCN(C(C2CCCCN2S(C)(=O)=O)=O)CC1 N1(C(CSCC#C)=O)CC(NC(C2(C)CCCN2C(C)=O)=O)CC(F)C1 C1(C(=O)OC(c2cccc([N+](=O)[O-])c2)CN(C)C)Cc2ccc(Cl)cc2S1 N1(C(COC2(C)CCOCC2)=O)CCC(C2CC2)C1CNC(c1cccnn1)=O C(=O)(C(CC)NC(c1ccc(CSC)s1)=O)NC(C1CN(CCC)C1)C c1(Nc2ncnc(N(C)C)c2Br)ccc([N+](=O)[O-])cc1S(C)(=O)=O O=C(NOCC1CCN1c1cn(C2CC2)nn1)C(F)c1ccccc1 C(=O)(CC(COC)NC(C1CN(C)C(=O)N1)=O)NC(c1ncnn1C)CC N1(C(C2OCCN(C(C(=O)NCC)=O)CC2)=O)CC(O)CC(C)(C)C1 OC1CCN(c2nccc(-c3ccccc3)n2)CC1O c1(C(N2C(CCC)CCC2)=O)coc2c1CN(C(c1cc(Cl)c[nH]1)=O)C2 N1(C(CS(C(C)C)(=O)=O)=O)CCCC2(CCC2NC(=O)COC2CCC2)C1 Cc1cn2cc(C(=O)NC(C)CNC(c3cnc(S)nc3)=O)cc(C)c2n1 CC(C)CC(O)C(=O)NCC1(C)CCCN(C(=O)CCc2cscn2)C1 C1(N(C(C(CC)OC)=O)C)CCCN(C(c2ccc(-c3ccccc3)cn2)=O)C1 N1(C(c2n(C)c(O)nc2)=O)CCC2CCN(c3ccc([N+](=O)[O-])cc3)CC2C1 c1(NC(C=C=C(C)C)=O)ccc2[nH]ncc2c1.N12CCN(CC1)C(=O)C2 CCCCCCC(C)(C)C(=O)NCCCC1CCCN1C(=O)CCC1CC1(C)C C1(NC(N2CCN(CC3(n4cccn4)CCOCC3)CC2)=O)CN2CCC1CC2 CN1CCC(O)(CC(=O)NC2CC3CC(NC(=O)CNC(=O)C4CC4)CC23)CC1 c1(C(=O)NC(C2CN(C(=O)C3=CCCCC3)CCO2)C)cnc2occc2c1 CCC(CC(=O)NCC(C(C)(C)C)NC(=O)CCc1ccc(C)c(Cl)c1)C(F)F c1(OC)ccc2nccc(NCC3(C(=O)C(CC(C)C)N)CC3)c2c1.C1(CO)CC1 c1(C(=O)NC(CNC(CCC(CC)C)=O)(C)CO)cnc2[nH]ccnc1-2 Cc1nc(C(=O)NCCC(=O)NC2CC23CC(O)C3)sc1C c1(CC)ccc(C(=O)NCC2(NC(=O)C(C)n3cncn3)CCOCC2)c(C)n1 CC1(C)C(=O)NCCN1C(c1cc(-c2ccc3c(c2)CCC3)on1)=O C1(CNC(CN2CCC(C)C2)=O)CN(C(=O)CC2=CCCC2)CC(C)(C)C1 CC1CC2(CCC2)CN1C(c1cc(CNC(C2CN(C)C2)=O)[nH]n1)=O C(=O)(N(CCCO)OC)C1CN(C(C(CC)(C)OC)=O)CC12CC2 C1(NC(Cc2cc(C)no2)=O)CCN(C(=O)Cc2sc(O)nc2O)CC1C C1(O)(CNC(C2C(CC)C2)=O)CCCN(C(=O)C(=CC2CCC(C)CC2)C)C1 Cc1cc(NC(C2CCN(C(=O)C(C)(C)C)CC2C)=O)ccc1SC(F)(F)F N1(C(CC(C)(C)C(F)F)=O)CCC2C(CCCN2C(c2cccc(O)c2F)=O)C1 C(=O)(C(C(C)C)C1CCC1)NCC1C(CNC(CCC=C(C)C)=O)C1 n1(CC)ncc(C(N2CCC(N(C)C(C3CN(C)CCO3)=O)C2)=O)c1Cl N1(C(CC(C(C)C)C)=O)CCCC2(C1)CN(C(C1(C(F)F)CCCO1)=O)C2 Cc1cc(C(=O)N(CC(C)NC(=O)C(CO)c2ccccc2)C)n[nH]1 C(=O)(C1CCCc2nnn(C)c21)NC(CNC(C(CSC)(C)C)=O)CO c1(NC(C2CCCCN2C(c2cc(Cl)c(F)c(Cl)c2)=O)=O)c(Cl)ccc(O)c1Cl N1(C(C(C)NC(CC)(C)C)=O)CCC(NC(=O)C2=C(Cl)CC2)C12CCCC2 Cc1cc(C(=O)NCC2(C)CCN(C(C34COCC3C4)=O)C2)nc(C)n1 C1(C(=O)Nc2c(CC(=O)OC)ccc(Br)c2)CC2CCC(C1)C2F C1(NC(CSCC(C)C)=O)CCN(C(c2cnc(S)[nH]2)=O)C1(C)C c1(N2C3C(NC(c4c(C)con4)=O)CC(CC3)C2)nc(Cl)nc(C)c1[N+](=O)[O-] CC(O)(CNC(=O)C(Cc1ccco1)NC(C1CC12CCC2)=O)CO C1(NC(c2c(OC)nn(C)c2)=O)CCC12CCCN(C(c1cnc[nH]1)=O)C2 N1(C(C2CCCN(CC)C2)=O)CCOCC(NC(=O)CCCN=[N+]=[N-])C1 Cc1ccc(C)c(C(=O)NCC23CC2CN(C(c2cnn(C(C)C)c2)=O)C3)c1N c1(C(=O)NCC2(F)CN(C(C3CCC(F)C3)=O)C2)cncc(C(F)(F)F)c1 c1cccc(CC(=C)CC)c1.c1(C2c3nnnn3N2)nc(CCC)cs1.OC N1(C(=O)NC2COCCN(C3CCN(C)C(=O)C3)C2)CCCOCC12CCCC2 C=CC(CCC)CC(=O)N1CC2CCC(NC(=O)Cc3c[nH]ccc3=O)(C2)C1 C123CCC1CN(C2)CC1(CCC1)NC(=O)C3.C1(C(=O)OC)CCC(N(C)C)C1 CCC(CNC(=O)CC1CCCC(C)O1)(CC)NC(=O)CCN1CCCCC1 CCCCC(N=c1[nH]c(C#N)c(Cl)s1)C(C)C(=O)NC(=O)Nc1ccccc1 Cc1cc(C)n2c(CNCc3cnoc3-c3ccccc3)nnc2n1 CCCCCC(CC)C(=O)NC(C1CCCN1c1ncc(Cl)c(O)n1)(C)C C1(C(N(CCCNC(c2c(C(C)C)n[nH]c2)=O)C(C)C)=O)CCCOC1C C1(C(=O)NC(CNC(C=CSC)=O)(C)C)C(F)(F)C12CC2 c1(OCC(N2C(CNC(COCCCC)=O)CC2)=O)cc(C(N)=O)ccc1CC c1(C(N2CC(OCCC(N3CCC(C)(C)C3)=O)C2)=O)cc(O)cc(=O)o1 N1(C(C2(OC)CCC2)=O)CCCC(CCNC(=O)CC2CCC(=O)NC2)C1 C(=O)(CC(C)CC(=O)NCC1CC2CCCC2N1C(=O)CC1C=CCC1)OC CC1CC(O)CN(C(c2cccc(C(C)(C)C)n2)C(=O)NC2CC2)C1 c1(OC)cc(C(N2CCC(C(C)NC(c3c(F)ccnc3Cl)=O)C2)=O)ccc1C C12(CNC(=O)Cn3nnc(=O)[nH]3)CN(C(c3cnc4n3CCS4)=O)CC1CCO2 N1(C(C(CC=C)OC)=O)CC2CC(O)C1C2NC(=O)Cn1cc(C2CC2)cn1 C1(NC(=O)C=Cc2ccsc2)CCCCC1NC(C1CCCCN1CC(F)F)=O c1(NC(C)C(=O)NC(C2(NCCO)CCCCC2)=O)cccc(SC(F)(F)F)c1 c1(C(=O)NCCn2cc(COC(=N)O)nn2)sc2cc(Br)ccc2c1Cl CC1CN(C(=O)CCCC(N)=O)CC(C)C1NC(=O)C=C(Br)Br N1(C(CC2(OC)CN(Cc3nn(C)cc3C)C2)=O)CC2CCC(CC2)C1 N1(C(C(CC#C)C)=O)CCC2C1CCCN2C(c1cc(=O)n(C)o1)=O c1(C(=O)NNC(=S)Nc2cccc(C(F)(F)F)c2)ccc2cccc(F)c2n1 N1(C(c2c(CC)noc2)=O)CC2CC1C2CNC(c1c(C)noc1C(F)(F)F)=O c1(C(N2C(CNC(C3CCc4c[nH]nc4C3)=O)C=CC2)=O)cc2cccnc2[nH]1 C1(C(N2CCC(Cn3cc(C(C(=O)OC)(F)F)nn3)CC2)=O)CCCCC(=O)N1 c1(C(N2CC(O)(CNC(CCc3onc(C(C)OC)n3)=O)C2)=O)cccnc1O c1(-c2c(CC)cccc2)ccc2cc(C(=O)Nc3cc(C)c(O)c(C)c3)cn2c1 C1(NC(C(CC)SC)=O)CCN(C(c2cnn3cc[nH]c(=O)c23)=O)CC12CCC2 CCCC(C)(CC)C(=O)NC1CCN(CCCNC(=O)CC2CCSC2)C1 C1(CCNC(=O)CCF)CC(F)(F)CN1C(=O)CC(O)C1CCCC1 CN1CC(NC(=O)C2=CCC(NC(=O)CCC3CCC(=O)C3)C2)C2(CC2)C1=O c1(C(N2CCN(CCOCCOC)CC2)=O)ccc2ncnn2c1 c1(C(=O)NCC2N(C(CCC=C)=O)CCC2C)ccnc2ccc(OC)nc12 N1(C(C(CC)C)=O)CC(NC(=O)CCc2ccccc2C(N)=O)C2CCCCC12 C1(C2CC2)(C(=O)NCC(C)(CO)CO)CN(C(=O)CN2CCNC2=O)C1 c1(CC(C(=O)NC(C(=O)OC)Cc2ccc(Cl)nc2)N)cc(Cl)c(O)c(Br)c1 N1(S(CC=C)(=O)=O)CCn2nc(C(=O)Nc3c(C)cccc3C)cc2C1 c1(CC(=O)NC(CC)CNC(C2CC(F)(CO)C2)=O)ncncc1Cl C1(NC(C(CC)OCC)=O)CN(C(c2cc(C)ccc2N)=O)CCC1(C)C c1(OC)ccc(OCC(=O)NCCCCN(C(=O)C(C)(C2CC2)OC)C)cc1 CC1(C2CCN(C(c3cn(CCNC(c4ccc[nH]4)=O)nn3)=O)C2)CC1 C1(NC(c2nc(C)oc2)=O)CN(C(C2(CNS(N)(=O)=O)CC2)=O)CC1O C1(CNC(c2c(C)cccn2)=O)N(C(=O)Cc2cc[nH]c2)CCCC1(C)C N1(C(c2c(C)nccc2)=O)CCC(C)(C)C1CC(=O)N(C)Cc1cc(=O)cc[nH]1 C1(CC)(CC)Oc2ccc(NCC3CCCN(C(=O)OC(C)(C)C)CC3)cc2O1 Cc1ncc([N+](=O)[O-])n1CC(=O)NCC(C)(C)CNC(C1CCCC1C)=O CCCCC(CNC(=O)C(C)(CO)OC)NC(=O)CCOCCCOC N1(C(C(CCC=C)NC(c2csc(=N)[nH]2)=O)=O)CCN(C)C(=O)C1C C1(CNC(CCN(C)CCO)=O)CC(O)C12CCC2.C12CC(CCO1)NC2=O N1(CC(C)NC(=O)C(CNC(C2CNC(=O)O2)=O)N(C)C)CCCC1=O Cc1ncccc1C(=O)NCCC(C)(C)CNC(=O)CCCc1nncn1C N1(C(C(CCC)C)=O)C(C)CC2CN(C(=O)COCCN(C)C)CC12 N1(C(C(C)N2CCC2)=O)CCN(C(=O)CN2C(=O)CNC2=O)CC1CCO Cn1cnc2c(NCC3(CC4CCC4)CC3)nc(N3CCOCC(CO)C3)nc12 N12CCCC(C1C)C2=O.Cc1nn(C(C)(C)C)cc1NC(=O)CSCCC(C)C C1(O)(CNC(C=Cc2n(C)cnc2)=O)CCCN(C(=O)CC(C)(C)O)CC1 C1(NC(C(=O)NC(c2c(Cl)ccc(F)c2Cl)C)=O)CNCC12CCCC2 CC1=C(C(=O)NCC2(NC(c3ccc(C(F)F)cc3)=O)CC2)C(=O)OC1(C)C O=C(CC1=CCCC1)NCC1(CNC(=O)C(F)(F)c2ccccc2)CC1(F)F N1(C(C2CC(C)N2C(=O)CCc2cccs2)=O)CCN(C)C(C)C1 C#CCC(C(=O)N1CCC(NC(=O)C=CC(=O)OC(C)(C)C)C1C(C)C)C1CC1 C(N=c1[nH]cnc(NCC(C)(C)S(C)(=O)=O)c1C)c1cncc(SCC)c1 c1(C(N2C(CN(C(=O)CN3CC4CC4C3)C)COCC2)=O)n[nH]c2c1COCC2 Cc1ccc(F)c(C(N2CCC(CNC(=O)C(C)(O)Cc3ccccc3)C2)=O)c1 N1(C(C2C(C)C2)=O)CCC(OCC2CCC(NC(=O)COCCF)C2)CC1 N1(c2nncc(OC)n2)CC(NC(c2ccc(N(C)C)cc2)=O)CC(C)C1 c1(CC)ccc(C(=O)NC2CC23CC(NC(=O)C(C)(C)CSC)C3)cc1 C1(C(N(C(C=C)C2CC2)C)=O)(NC(C2CCCN2C(=O)OC)=O)CC(F)C1 c1(OCC)ccc(C)nc1C(=O)NCC(C1CCC1)NC(=O)C(C(C)C)NC=O c1(C(N2C(CN(C(CSCC=C)=O)CC)CCC2)=O)cc(N)ccc1C N1(C(C(C)N2CCCC2)=O)CC2CCCC2C1C(N1CCCC(O)C1C)=O c1(CNC(=O)CC2CCCCCC2)ccc(C(=O)NC(CN(CC)CC)C)cc1 CC1CN2CCN1CC2C(=O)NC1(CCNC(=O)CC2CCCSC2)CC1 C1(CNC(c2cc(CC(C)C)[nH]n2)=O)(NC(=O)C(O)C(C)C)CCC(F)(F)CC1 c1(C(=O)NCCC(C(=O)NC2CCN(CC)CC2C)(C)C)cccc(C)c1C#N C1(NC(C2CCC(N(C)C)CC2)=O)CN(C(=O)Cc2cccc(F)c2)CC12CC2 N1(C(C(CO)OC)=O)CCOCC1C(=O)NCCc1cnc[nH]1 N1(C(CNC(CCc2n(C)cnn2)=O)=O)CCCCC(CO)C1 N1(C(C(C2(O)CN(C(C(C)CC(F)F)=O)C2)F)=O)C2CCC1CC(F)C2 CCCC(C)C(=O)NC(C)CCN(C)C(C1CC1c1cnn(C(C)C)c1)=O n1(CC(=O)N(CCC)CCNC(=O)C(O)Cn2cncn2)cnc2c1CCCC2 N1(C(C(C)SC)=O)CC(NC(c2cscc2SC)=O)CC1(C)C C1(CC(=O)NCC(CC)NC(=O)C(C)(C)CSC)SC2=NCCN2C1=O N1(C(Cc2c(COC)cccc2)=O)CCOCC(NC(C2(C)COC2)=O)C1 N1(CCC(=O)N(CCOCCN(C(CS(CC)=O)=O)C)C)C(=O)NC(C)(C)C1=O N1(C(C2C(C(=O)OC)C2)=O)CC(C2CCCN(C(=O)CCCC3CCCC3)C2)C1 C(CCCC(CO)NC(=O)C(C)c1cc[nH]n1)NC(c1c(C(C)C)cccc1)=O N1(C(C(CC)C)=O)CCC2CN(C(c3cc4cc(Cl)ccn4n3)=O)CCC12 CC(C)CC(C)(CNC(=O)C(c1ccc(F)cc1)CO)NC(=O)C(=O)NC1CC1 Cc1ccc(F)c(CC(=O)NC2(C)CCCN(C(=O)C=Cc3sccc3C)C2)c1 C1(C(=O)NCC2(F)CC(NC(=O)CC3(O)CCC3)C2)CCCOC1c1cc[nH]n1 CC(C)CC(F)(F)C(=O)NCC(C1CC1)N(C(=O)C(C)Cc1ccc(F)cc1)C N1(CCC(=O)NCC(C2CC2)NC(c2c(CC)nns2)=O)C(=O)NC(C)(C)C1=O C(CC(C(=O)NOC1CCCC1)NC(=O)C(C1CCCC1)OC)OC C=CC1COCC1NC(C12CC(CO1)C2)=O N1(c2c(C)cc(C3CC3)cn2)CCc2nc(N3CCN(C)CC3)ccc2C1 N1(C(c2c(CC)ccs2)=O)C2CCCC1CN(C(c1cc(C(C)C)n(C)n1)=O)C2 c1(C(=O)NC2CCC(CC(=O)N(CCN=[N+]=[N-])C)C2)cc2ccccc2o1 C(=O)(CCCCC(=O)NCC1CC(C)N(C(=O)CCc2nc(C)cs2)C1)OC C12(C)CN(C(C)(C)C1)C2=O.c1(CNC(c2c(CC)cc[nH]2)=O)cccc(O)c1F CC(CC(=O)NCC1(O)CCN(C(=O)CCN2CCCCC2C)C1)CC(C)(C)C Cc1nc(C)n(CC(=O)NCc2ocnc2C(=O)NC23CC(C2)C3)n1 C(C)(C(=O)N1CC(CC(N2CC(OCC(N)=O)C2)=O)C1)OC(C)=O c1(OC)cc(O)c(OC)cc1Oc1ccc(Br)cc1CN1CCC(OC)C1 N1(C(C2C(=C)C2)=O)CCC(CO)(NC(=O)COCc2ccccn2)C1 C1(C)(NC(C2CN(C)C(=O)C2)=O)CCCN(C(=O)Cc2c[nH]nc2O)C1 C1(NC(Cc2c(C)noc2C)=O)CC(NC(c2cc(C)n(C)c2C)=O)C12CCC2 C1(N(C(=O)C(F)OC(F)(F)F)C)CN(C(=O)Cc2csc(=N)[nH]2)CC1F C(=O)(C(C)(O)C(C)C)N1CC(CC=C)(NC(=O)C(N2CCSCC2)C)C1 C1(C)(NC(CC2C(CNC(c3c(CC)cccc3)=O)C2)=O)C(C)(C)C1(C)C c1(C(N(CCC)CC2CCCO2)=O)cn2c(n1)CCN(CC1CC=CCC1)CC2 C12(C(=O)NC(C)CN(C)C(C3CCC3C(C)(C)C)=O)COCC1C2 CC1(C)C(C(=O)NC2CCN(C(=O)CCCc3nncn3C)C2C2CC2)C1(C)C c1(-c2cn(CC3C(NC(CCc4cnn(C)n4)=O)CCC3)nn2)cncc(N)c1 c1(C(N2CC(NC(=O)CC3CCCCC3O)C3(C2)CC3)=O)ccc2nncn2c1 c1(C(=O)NC2C(CNC(=O)Cn3nnc(C(F)(F)F)n3)C2)ccnnc1S C1(C(N2CCN(C)C(=O)C2)=O)CN(C(C2CCS2(=O)=O)=O)CCC1(C)C c1(OC)ccc(C(O)C(=O)N(C2CCN(C(c3c(C)n[nH]c3C)=O)C2)CC)cc1 C1(NC(C2ON=C(C)C2)=O)C2CC1CN(C(c1ccccc1C(F)(F)F)=O)C2 C1(N(C(c2c(C)nns2)=O)C)CCN(C(C)C(=O)NCc2ccccn2)CC1C C1(CNC(CCNC(CC2C(CC)C2)=O)=O)CCCC1(C)C CCC(C)C(C)C(=O)NCc1ccccc1CN(C)C(c1ncnc(C)c1C)=O C1(F)(CC)CCN(C(=O)CC2CC(NC(=O)C=Cc3cc[nH]c3)C2)C1 c1(C(=O)NCCC(CCC)C(=O)OC)cnc2c(F)c(F)ccc2c1 C1(C(=O)NCC2(F)CCOC2)(NC(Cc2c(C)n(C)nc2)=O)CCC(C)(C)C1 C=CC1(C(=O)NCC2(OC)CN(C(=O)CC(C)c3ccccc3)C2)CCOCC1 c1(C(N2CC(C)C(NCc3cc(F)c(Cl)cc3O)C2)=O)cccc([N+](=O)[O-])c1F N1(C(C(=O)NCC)C(C)C2CCCC2)CCN2CC(O)CC2C1 C(=O)(CC(C)(C)C(=O)NCCC1CN(C(=O)C(C)OCC(C)C)CCCO1)OC N1(C(C(c2cc(C)sc2)(F)F)=O)CCC2(NC(=O)Cc3ccnn3C)CCCC12 N1(C(C=COCC)=O)CCCC1(CNC(c1c[nH]nc1C)=O)COC c1(NC(c2nnnn2CC2CC2)(C2CCCOC2)COC)cc(Br)ccc1C CCC(CCCC(=O)N(C(C)CN(C)C)C)NC(=O)C=Cc1cncs1 C(=O)(C(CCSCc1cscn1)NC(=O)OC(C)(C)C)N(CCOC)C C12(NC(Cc3nc(C)sc3C)=O)CCCC1CN(C(=O)C=CC1CCOC1)C2 C=CCC(C)(C)CC(=O)OCC1NC(=O)NC1=O.c1(C(=O)NCC)cscc1 c1(C(C)(C)C)cn2c(n1)C(C(=O)NC13CC(NC(=O)CCC(N)=O)(C1)C3)CCC2 N1(C(CC=C(C)C)=O)CC(C)OC2(CCN(C(c3nnn(C(C)(C)C)n3)=O)C2)C1 C1(c2cc(C)on2)CCCN1N1CCC(C(C)(C)O)C1 CC(C)CCC(F)C(=O)NC(C(=O)NC1CCCC(C2CC2)C1)C1(C)CC1 CN1C2CCCC1C(N1CCN(C(C3CC4(CCN4)C3(C)C)=O)CC1)C2 Cc1c(NCc2nccn2C2CC2)ncnc1N(C)Cc1nccn1C(F)F C(=O)(CC(C)CC(C)(C)C)NCC1(F)CCC(NC(C2(COC)CC2)=O)C1 N1(C(CSCC#C)=O)CCC2(CCCN2C(=O)COCC2CCCO2)C1 c1(C(N2C(C)CC(CNC(C3(O)CCCC3)=O)C2)=O)coc2c1CCCC2 c1(C(=O)OC)ccc(-c2cncnc2N2CC3CC(O)C2C3)cc1F c1(C(N2CC(CNC(=O)Cn3ccnn3)C(O)C2)=O)ccnc2ccc(F)cc12 c1(C(C(N)=O)NC(=O)NCc2cccc(C(F)(F)F)c2)ccc(Cl)cc1F C1(C(N(CC(c2nn[nH]n2)C)C)=O)CC2CCCC2N1C(C1C=CCCC1)=O C#Cc1cc(C(=O)NC2CCN(C(c3ccc(CC)s3)=O)C(C)C2)ccc1Cl S(=O)(=O)(c1cccc(C#N)c1)N1CC(NC(Cn2c(C)c(Br)cn2)=O)CC(F)(F)C1 N1(C(CSCC=C)=O)CC(N(C)C)C(CNC(=O)C=C(Cl)Cl)C1 C1(CCC)CN(C(C2(C#N)CCCOC2)=O)CCN1C(=O)Cc1ccccc1Cl C(CC1OCCc2ccccc21)NC(=NCCOCC)NCc1cnn(CC)c1 c1(C(=O)NC(C2CN(C(=O)CC3C=CS(=O)(=O)C3)C2)C)cnc(C2CC2)nc1 c1(-c2nnc(SCC(=O)NCCC(C)NC(C=C(CC)C)=O)o2)ccc(F)cc1 c1(C(N)=O)cc(C(=O)NCC2CCCN2C(c2ccnc(Cl)c2)=O)ccc1O Cc1ccc(O)cc1C(=O)NNC(=O)NC(c1cncn1C)C1CCCC1 c1(C(=O)NC(C2(O)CN(C(C(C)SC(C)C)=O)C2)C)cc2n(c1)CCCC2 Cc1cc(C(=O)NC2CC2NC(c2cncc(Cl)c2)=O)ncc1S(N)(=O)=O Cc1cc(Cl)c(C(C)NC2CCN(CCCO)CC2)cn1 N1(C(CC=C=C)=O)CCC(C)(C)C(C(=O)NCc2nc(C)no2)C1 c1(C(=O)NC(C(=O)NCCC(C)SC)C2(O)CCC2)ccc(CF)cc1 Cc1cc(C(=O)NCc2cc(C(N3CCCCC3CN(C)C)=O)n[nH]2)c(C)nn1 N1(C(=O)OCC)CCC2(CC1)CC2(C)NCCS(=O)(=O)N(C)C C1(NC(Cc2cccc(OCC)n2)=O)CC2CC(NC(=O)CNC(=O)CC)C2C1 C1(C(N2C3C(NC(C4N(C)CCC4)=O)CC(CC3)C2)=O)CCCC12CCOCC2 c1(C(=O)NCC2CC(O)CN2C(C2CCCS2)=O)noc2c1CCCC2 N1(C(CCCN(CCC)CCC)=O)CCC2CC1CN(C(=O)CNS(C)(=O)=O)C2 CCC(C(=O)N1CCC(N(C(=O)CCCOCC)CC2CC2)CC1)C(C)O CCCC(C)(CC)C(=O)OCC1(C)CCN(CC2CCC(C)CC2)CC1 O=C(CC1=CCCCC1)NC1CC(CNC(C2(c3ccno3)CCOCC2)=O)C1 Cn1cc(NC(=O)CCC2CCN(C(=O)CCn3ccnn3)C2)c(C#N)n1 N1(C(c2n(C)ncc2Cl)=O)CC2(CCN(C(C3CN4CCCN3CC4)=O)CC2)C1 N1(C(C(CCNC(C(C)NC(=O)NC)=O)(C)C)=O)CC2CSCC2C1 c1(C(N2CC(CC=C)(NC(c3cc(C4CC4)ncn3)=O)C2)=O)nccc(Cl)c1C C1(C2CCC2)(C(=O)NCC(C)(C2CC2)NC(C2CCCC(=O)O2)=O)CCCCC1 c1(NCCc2[nH]nc(O)n2)nc(N2CCC(CC(F)F)C2)c2c(n1)COC2 c1(C(N(C2CCN(C(c3nc(=O)n(C)[nH]3)=O)CC2)C)=O)cnc2ccncc2c1 C1(NC(c2c(CC)nc[nH]2)=O)CCC2CCN(C(=O)C(c3ccc(C)s3)C)C12 c1(C2N(C(=O)NC3CCN(c4ccccc4)C3)CCC2)ccc(F)cn1 C1(NC(C(C)(C)C)=O)CCCCC1CNC(c1ccc(-c2cc(O)ns2)cc1)=O N1(C(CC2CN(C(CN(CCCC)CC)=O)C2)=O)CCCC(OC2CC2)C1 N1(C(c2c(CC)csc2)=O)CCC(NC(c2nc(OC)c(C)s2)=O)CC1C CCC(CC(=O)NCC1(O)CCN(C(=O)CCN2CCC2)C1)C1CC1 c1(C(=O)NC23C(CN(C(C4C(C=C)CC4)=O)C2)C3)sccc1S(C)(=O)=O c1(C(=O)NCCC2(C(=O)NCC(C)Nc3ccsn3)CC2)ncccc1C1CC1 N1(C(c2cc(C(NC(=O)C(c3cccnc3)O)CCO)[nH]n2)=O)Cc2ncsc2C1 C(C(=O)N=c1cc(-c2cccnc2)[nH][nH]1)(c1cccc(OC)c1)SC c1(C(N(CC(C)C#N)CC)=O)ccc(SC(C)C(=O)OC)cc1 C#Cc1cncc(C(=O)NCC2COCCN2C(c2ccc(CO)cc2F)=O)c1 Cn1ccc2c(C(=O)NC3CC34CCN(C(=O)COC(F)(F)F)CC4)ncnc12 C1(NC(C(C)OCC=C)=O)COC2(CNC(=O)CCCCc3cnc[nH]3)CC1C2 C1(C(=O)NCC2(C(=O)NC(CCC=C)C3CC3)CCC2)C2CCC(F)(F)C12 C(C(CC(F)(F)F)NC(c1ccsc1OC)=O)NC(C(CC)SC)=O c1(CNCC2CCN(C(c3cncn3C(F)(F)F)=O)C2)cc(Cl)sc1Cl Cc1ccc2c(c1)N(C(=O)CC1(NC(C3CCCN3C=O)=O)CC1)CC2 CCC(CC)CC(F)C(=O)NCc1nocc1C(=O)NCc1cc(C)on1 c1(NC2C(SCC)CCC2)[nH]c(=NCCN2CCCCC2=O)nc2scnc12 Cc1c(NCc2ccccc2Cl)nc[nH]c1=NCC12CC(C)(CCO1)C2 c1(C(=O)NC(C(N2CC(OCC)C2)=O)c2cccs2)ccc(O)c(F)c1F Cc1ccc(F)cc1CN(C)CC1CN(C(c2cccc(Br)c2O)=O)C1 Cc1c(C(C(C)C)NC(c2cncc(N(C)C)c2)=O)oc2ccccc12 Nc1c(Cl)ccc(F)c1C(N1C2CCC1C(NC(c1cnc(C3CC3)o1)=O)C2)=O c1(C(=O)NC)c(C)[nH]c(C(=O)N(C(C)C(C)(C)C)C)c1C N1(Cc2scc(C)n2)CCN(C(c2csc(CCP(C)(C)=O)n2)=O)CC1 N1(C(C(C(=O)OC)C)=O)C2CCC1C1CC1(NC(=O)CCc1cccc(C)c1)C2 C1(C(=O)NC(CNC(Cc2cccc(OC)c2)=O)C(C)C)CCC(C)(C)CC1 C=CCN=C(NCCC(C)(C)COC)NCC1(C(F)(F)F)COC1 Cc1csc2c(C(=O)NC3(C4CN(C(C5(C)CCOC5C)=O)C4)CC3)cccc12 c1(Nc2cccc(-c3scc(C)n3)c2)nccn2nc(C(=O)O)cc12 N1(C(CCCCOC)=O)C2CCCC1CC(NC(c1cc(C(C)=O)c(C)o1)=O)C2 Cc1ccc(C(CNC(C2CC2(Cl)Cl)=O)NC(c2ccn(C(C)C)c2C)=O)cc1 c1(C(N2C(CC(=O)OC)CC3(CC3)C2)=O)csc(S(C)(=O)=O)c1 C=CC(F)(F)C(=O)NCC1(F)CN(C(c2cnn(CC3CCCC3)c2)=O)C1 C=CCN(Cc1ccccc1)N1CCC(CCOC)C(F)(F)C1 C(=O)(C(C)(C)C(O)C(C)C)N1C(C(=O)OC)CC(Oc2cccc(OCC)c2)C1 c1(CC)nc(C(N2CCCC2C2CCN(C(c3cnsc3)=O)C2)=O)c(N)s1 C1(CNC(COCC(=C)C)=O)CC2CC1CN2C(C1C=CCC1)=O N1(CC(=O)NC(C2CCCCC2)CC)CCCCC1Cc1cccc(C)c1 c1(C(=O)OC)ccc(C(=O)NC2(C(=O)O)CCC2)cc1OC c1(CCC(N2CC(NC(c3n(CC)ccc3)=O)C3C2C3)=O)c(O)nc(=N)[nH]c1C c1(SC(C)C(N2CCN(C(=O)CP(C)(C)=O)C(C)C2)=O)ccc(C#N)cc1 C1(C(=O)NC(CC2CCOCC2)C(N2CCC23CCCC3)=O)CCC2(CCC2)O1 c1(C(N2CC(COC)(NC(c3cccnc3C)=O)C2)=O)cccn2c(O)nnc12 C1(C(=O)NCCC2(O)CN(C(C(C=C)O)=O)C2)(C(=O)OC(C)(C)C)CCSCC1 Cc1ccc2c(c1)OC2.c1(C(=O)NCc2cccnc2)c[nH]nc1Cl C1(CNC(c2ccc(C)nn2)=O)COCCN(C(c2cncc(Cl)c2C)=O)C1 c1(-n2c(-c3coc(C4CC4)n3)nc(CCCN(C)C)n2)cc(Cl)nc(Cl)c1 c1(OC)ccc(CN(C(=O)NC2C3CC4C(C3)C24)CC2CCCSC2)cc1 c1(C(C)NC(C(COC)NC(=O)C(O)Cn2cncn2)=O)c(C)n[nH]c1C C1(CNC(C(COC)(C)C)=O)CC2CCC1N2C(c1cncc(C(C)C)c1)=O O=S(=O)(c1ccc(-c2csc3ccccc23)cc1)NCCc1cccc(F)c1Cl C1(C2CC2)(C(N2CC(CC(COC)(C)C)C2)=O)CN(C(C2C3CCCCC23)=O)C1 N1(C(c2cc(C)n(C)c2)=O)CC2CC(NC(c3nncn3C)=O)C2C1 CC1(O)CCCN(C(=O)NCC2CCC=CCCC2)C1 N1(C(C=COC)=O)CCOC(C(C)NC(c2cnccc2N(C)C)=O)C1 S(=O)(=O)(c1ccc(NCC(C)OC)nc1)N(C(CCCC)(C)C)CC C1(NC(CC2N(C(C(C)(C)SC)=O)C3C2CCC3)=O)CCN2CCCC2C1 CC(C(=O)N1CC(F)(CNC(C23CCC(F)C2CC3)=O)C1)S(C)(=O)=O CS(=O)CCC(O)C(=O)N1CC(O)(CCNC(c2cc(Cl)ccc2N)=O)C1 C1(NC(=O)NCc2cc(C)nn2C)CCCC(OC(C)(C)C)CC1 C1(NC(CC=CC=C)=O)CCN(C(=O)C(C)(C)C(C)C)CC1(C)C Cc1cccc(F)c1CC(N1CC2CC1C2NC(=O)Cn1nnnc1C)=O N(C(=NCCc1ccc(O)cc1)NCC(O)COC1CCOC1)C(C)CC1CC1 N1(C(c2cnc3ccnn3c2)C(=O)NC(CC)(C)C)CCCN2CCCC2C1 C1(C(=O)Nc2ncc(C(C)(C)C)[nH]2)CN(C(c2cc(Cl)sc2Cl)=O)CCC1O n1(CC)nc(C)c(C(=O)NCC2CCC(NC(C3CCSC3)=O)C2)c1Cl c1(CC(=O)NCCN(C)Cc2cn(-c3ccncc3)nn2)ccc(S(N)(=O)=O)s1 N1(C(C=C(COC)C)=O)CCCC(CCC(=O)NC(CCO)C2CC2)C1 c1(C(N2CC(NC(c3c(Cl)cnc(SC)n3)=O)C(F)C2)=O)cc(Br)cc(Br)c1O n1(CC)nnnc1C(C)(C1CC1)NC1(c2cccs2)CC1 C(=O)(C1Cc2ccc(Cl)cc21)NCCN(C(c1c(CC)con1)=O)CCOC c1(C(N(CCCNC(c2ccn(CC)n2)=O)C2CC2)=O)cc(Cl)c(OC)cc1Cl Cc1c(C(=O)NC(CNC(c2cccnn2)=O)C(C)C)ccc2c1OC(F)(F)O2 NS(=O)(=O)CCCC(=O)NCC1CC(NC(C2CC3CCC2CC3)=O)C1 CC(CC1CCOCC1)C(C(=O)NC1CCOC1)N(C1CCN(C)CC1)C N1(C(c2cc(-c3ccc(OC)c(Br)c3)no2)=O)CCC2(CC1)CCS(=N)(=O)C2 C#CCC(CC(=O)N(C)CCn1cncn1)NC(=O)C(CCCC)N(C)C C(c1cccnc1)=C(C)C(N1CCC(C)(NC(=O)C(F)=CCCF)C1)=O Cc1c(CCC(=O)OC(C)(C)C)cccc1Br N1(C(Cn2c(C)c(Cl)cn2)=O)CCC(CCNC(c2cn(C)c(O)n2)=O)CC1C C(CS(=O)(=O)CCN=c1[nH]c(=NCC(C)OC)[nH]c2c(F)cccc12)OC C1(NC(CC(=C)Br)=O)CC2(CCN(C(=O)CCC(C)N(C)C(C)=O)C2)C1 Cn1cc(C(=O)NCC2C(CNC(=O)CN(C3CCC3)C)C2(F)F)ccc1=O C=CCC(CNC(c1ncccc1Cl)=O)C(=O)NC(CC(=O)NC)C1CC1 C(=O)(CC(C(F)(F)F)NC(c1coc(CO)c1)=O)N1CCCC(C)(CO)C1 Cc1ccc(C)c(C(N2CCC(CF)(NC(=O)CC3CC=CCN3C)C2)=O)c1N C1(C(=O)NCC(=C)Br)CN(C(=O)Cc2nc(=N)[nH][nH]2)CCC1(C)C N1(C(CC(CNC(C(=O)NCC)=O)OC)=O)Cc2ccccc2C1 C1(NC(CC(=C)C)=O)CN(C(c2nc(C(F)(F)F)ccc2Cl)=O)CCC1C Cn1cc(SC=CC(C)(C2CCC2)NC(=O)C(=O)NC(=O)C=CBr)cn1 N1(C(Cc2cccc(C)c2)=O)CCN(C(c2cc(O)nc(Cl)c2)=O)CC1C Cc1ncc(Br)c(N2CCC(NC(c3ncn(C)n3)=O)C(O)C2)n1 N1(C(Cn2nnc(C)n2)=O)CC2(CCN(CCCC(C)(C)C)CC2)CC1C CCCCCC(CC)C(=O)NCC1CC(F)CN1C(c1ccn2c1CCCC2)=O C1(C)(C(=O)NC2CCC(CCC(=O)NCC(C)(O)C3(C)CC3)C2)CC2CC2C1 C(=O)(C(CC(C)C)ONC(=O)CC(C)ONC(c1cc(CO)on1)=O)OC N1(C(C=C(CC)C)=O)CCC2(CC1)CC2CNC(C1CC2CCC1C2)=O C(=O)(C(F)C(F)(F)F)NC1C(NC(c2onc(OC)c2Br)=O)CC1 c1(C(N(C2CCCC2)CCCNC(C2OCC(C)C2)=O)=O)cnc2occc2c1 N1(C(C2CC(CC)NCC2)=O)CCC2(CCCNC2)CC1 Cc1c(C(=O)N(C)CC2CCCN2C(=O)CCCC2CCCC(=O)N2)ccn1C c1(CNC(=O)NC(c2cccc(OCC)c2)CCC#C)cc(N)ccn1 C1(C(C(=O)NCC2CCOC2)N(CC(F)F)C(C)C)CCCC(C)C1 C(=O)(C1=CCCC1P(C)(C)=O)N1CCC(C)(NC(c2c[nH]nc2C2CC2)=O)CC1 C1(C(N2CCC(C)(C)C2)=O)CC2(CCN1)CCOCC2 c1(OCCC(=O)OCC2(CCOC(C)C)COC2)ccc(F)c(F)c1 c1(CNC(c2c(C)cno2)=O)ccccc1CNC(=O)CC1CC(CF)C1 c1(C(=O)NC2CN(C(COCc3nnc(C)s3)=O)CC2O)nc(F)ccc1Cl N(C(=NCc1cccc(Cc2n(C)ccc2)c1)NCC(Cl)C(F)(F)F)CC1CC1 C1(C(=O)NCC2(CCNC(C(C(C)C)O)=O)CC2)CCc2ncnn2C1 n1(CC(=O)NCCCCCNC(C2CC(=C3CCC3)C2)=O)ncc2ncccc12 N1(C(CCC(CC)C)=O)CCC(C2CC2)(CNC(c2ccon2)=O)C1 c1(OC)cc(F)ccc1C(=O)NCC1CN(C(=O)Cc2ccc(Cl)s2)CCCO1 N1(C(C(C2CCCCC2)OC)=O)CC2CC(NC(C3(C)CC3)=O)CC(C2)C1 c1(C(=O)NC(C(=O)N2C(C)(CC)CC2)CCOCCO)ccc(C)c(O)n1 C(=O)(C1=C(C#N)CCC1)NCC(C1CCN(C(C(CC(C)C)C)=O)CC1)(C)C C1(CNC(C(C)N2CCC2)=O)CN(C(=O)Cc2cccnc2F)CC(C)(C)O1 c1(COC(C(Cc2cccc(C)c2)C)=O)c(F)c(F)cc(C)c1F c1(C(=O)NC2CN(C(c3c[nH]nc3Br)=O)CCC2O)cc2cncn2c(O)n1 c1(CCNC(C2(CCCOC)CCCC2)=O)cc(Cl)sc1Cl C12C3CC(CC13)C(=O)N2C.N1(C(=O)OC(C)(C)C)CCCC1c1cccnc1 C12(NC(C3CCC(CC)O3)=O)COC(CNC(c3cc(C4CC4)on3)=O)(C1)C2 C(C(C(=O)N1CCc2nn[nH]c2C1)C(C)(C)C)NC(C(COC)N(C)C)=O c1(-c2cn(C)nc2)nc(CC2CCCC2)nn1-c1ccnc(O)c1 C1(C(N2C3C(NC(C(CCCC)(C)F)=O)C(C3)C2)=O)CCn2c(cnc2C)C1 c1(C(N2C(CNC(CNC(=O)OC)=O)COCC2)=O)cc2nc(Cl)ccc2s1 C1(C(=O)NCC(CC)NC(c2cnc[nH]c2=N)=O)CC(c2ccccc2)=NO1 c1(OCC(=O)NCCNC(c2cc(Cl)no2)=O)ccc(Cl)cc1 NS(=O)(=O)c1cc(C(=O)N(CCCNC(C2(C(F)F)CCCC2)=O)CCO)cs1 CC(c1ccccc1Cl)=CC(=O)NCC(C1CCC1)NC(c1ncsc1C)=O CN=c1[nH]nc(CC(N2CCC(CNC(c3c(C)ncn3O)=O)CC2)=O)s1 C1(CN(C)C)CCCN(C(c2cnn(CCNC(=O)CN3CC4CC4C3)c2)=O)C1 C=CCC(CC)C(=O)N(CCSc1cc(C(=O)N(C)C)no1)CCOCCO N1(C(c2noc(CC)c2C)=O)CCC(C2CC2)C1C(=O)NC1(C)C(C)(C)C1(C)C C1(C(Cn2cc(CSC)nn2)F)CCN(C(c2c(Cl)nsc2Cl)=O)CC1 C1(CCNC(=O)CCNC(c2cccs2)=O)CCCN1C(c1ccsc1)=O C1(C(N2C(C(N)=O)CC2)=O)COC2(C1)CN(C(=O)C=Cc1ccc[nH]1)C2 N1(C(c2cc(C)c(C)o2)=O)CCC2(CCN(C(C3CCC(C)NC3=O)=O)CC2)C1 c1(C(N2CC(NC(C(CC)(C#N)CC)=O)C(C)C2)=O)cncc2ccc(F)cc12 c1(C(=O)NCCN2CCN(C(C3C(C)C3)=O)CC2)ccc2c(c1)OCCCO2 Cc1ccccc1CCNC(=O)C=CC1CCCN1C(=O)C(C)O n1(CC)ncc(Cl)c1C(=O)NCC1(C(C)(C)C)CCN(C(=O)C(F)=CC2CC2)C1 N1(C(C(C)C2CC2)=O)CCC(F)C(NC(c2cnc(N3CCOCC3)nc2)=O)C1 c1(OC)c(C(=O)NC2CN(C(=O)C3=CCCCO3)CC2F)cccc1[N+](=O)[O-] c1(C(=O)NCC2(C=C)CCC2)cccnc1NC(=O)C(CC)NC(=O)C1CC1 C(C1(CC(=O)OC)CCOc2ccccc21)NC(CC(C(=O)OC)(C)C)=O CC1CC(NC(C2CC23CC3)=O)CN(C(=O)C#CC(=O)N(C)C)C1 C(C(=O)NC1CCOCC1)(C(C1CCCC1)OC)N(CCCN(C)C)CC CCC(CC)(C(=O)NC1CC1NC(=O)CSc1ccc(F)cc1)OC C(=O)(C(C(C)C)NC(C1(F)CC=CC1)=O)NCc1c(C)nn[nH]1 c1(C(N(CC(CN(C(CSSC)=O)C)O)C)=O)ccc2cc(C)ccc2n1 CCC(C)C(C(C(=O)NCc1ccco1)N1C2CCCC1COC2)OC Cc1cc2c(cc1C)N(C(C1(C)CC3(CCC3)C1)=O)CC2 S(=O)(=O)(c1ccc(-c2cccc(O)c2)cc1)N(C1CC(F)(F)C1)C c1(C(=O)NC2CN(C(CC3(C)CCCCC3)=O)C2)cc2nc(F)ccc2o1 CN1C(=O)CCC1C(=O)NCCN(C(C1CCOC1)=O)Cc1cccc(Cl)c1 c1(C(C)NC(=O)OC(C)C)cccc(NC(=O)C(=O)NCC2CC3(CC3)C2)c1 Cc1nc(C)n(CCCC(=O)NC2CCN(C(c3coc(C(F)(F)F)n3)=O)C2)n1 c1(C(=O)NCCN(C(=O)C(C)C2CCCC2)CC)cc(=O)c2ccccc2n1C C1(CNC(C=C(CCC)C)=O)CCCCN1C(=O)COc1cc(C(F)(F)F)ccn1 N1(C(CCSC)=O)CC(C)CN(C(c2cnc(CO)nc2C)=O)CC1C c1(NC2CC(CC(C)(C)C)C2)ccccc1CCP(C)(C)=O C(=O)(CCC(C)S(C)(=O)=O)N1C(CN(C(C(CC=C)(F)F)=O)C)CCCC1 CC1CC(C)(C(=O)NC2CCN(C(=O)COCCN(C)C)CC2CO)CCO1 c1(C(N2CCN(C(c3nccc(CC)c3)=O)C(C)C2)=O)c(C)cc(C)cc1O N1(C(CCSC)=O)CCN(C(=O)C(C2CCOC2)OC)CC(C)C1 N1(C(C2N(C(CCC)=O)CCC2)=O)CC(NC(C2CCCN2C)=O)CC(F)(F)C1 C12(C(N3C(C)CC(F)C3)=O)CCC(NC(C3CCC(N=[N+]=[N-])C3)=O)(CC1)CC2 C1(NC(=O)CC2CC2(Cl)Cl)CCCC1NC(C1CCCN1c1nccs1)=O Cc1ccccc1OCC(=O)NC1(CNC(C2(c3ccncc3)CC2)=O)CCC1 C12(CC(=O)NC(C(=O)OCCCC)C)CCC1CN(C(=O)CCn1ccnn1)C2 Cc1conc1CNC(C1CCCC1CNC(C1CCC1C(C)(C)C)=O)=O c1(OCC)ncc(C(=O)NCC2CN(C(c3ccsc3Cl)=O)C3CC23)cc1Cl N=c1cc[nH]cc1C(=O)NC1CCN(CCNC(=O)Cc2ccccc2)CC1 CC1(C(N2CC(c3ccc(F)cc3)C2)=O)CCN(Cc2ccccn2)CC1 C(C(CC(F)(F)F)NC(=O)CC12CCCC1C2)NC(c1cncc(C(C)C)c1)=O C(=O)(CC(=O)NC(C)CC(C)NC(=O)C(C1CCCC1)NC(C)=O)OCC CCC(Cc1ccccc1)CC(=O)NC1C2(NC(C3(CO)CC3)=O)CCC(C1)C2 c1(C(CNC(=O)CNC(c2ccn(C)n2)=O)OC)ccccc1C c1(C(N(C)Cc2nc(N3CC(c4ccccc4)C3)sn2)=O)cc(O)nn1C C(=O)(CCC(CF)CF)NC(c1ccccc1)C(=O)NCC1(O)CCC(C)C1 c1(CCC(=O)NC(C2CCCCC2)C(=O)OCC)c[nH]c2ccc(C)cc12 C1(CNC(Cc2cccc(CC)c2)=O)CN(C(=O)CC2(C)CC2)C2CCCC2O1 c1(C(=O)Nc2cccc(F)c2C(N2CC3CCC2C3)=O)cc(Cl)cc(Cl)c1O N1(C(C2OCC(C)C2)=O)CC2CCCN(C(c3ccc(-c4ccco4)o3)=O)C2C1 CC1(CNC(C2(C#N)CC2)=O)CCC(NC(c2csc(C(N)=O)n2)=O)C1 c1(OC)cc(OC)c(F)c(CN2CCC2C(=O)NC2CC(CO)C(O)C2O)c1F CC12CCCC(C(N3CCC(CNC(=O)C=Cc4ccc(F)cc4)C3)=O)(CO1)C2 c1(C(C)NC(c2csc(-c3ccccc3)c2)=O)ccc(O)nn1 c1(C(=O)NCC2CN(C(C(c3ccccc3Cl)(C)N(C)C)=O)C2)nnccc1C C1(C(=O)Nc2ccc(C(=O)OC)cc2C)CC2(C1)NCCN1CCCC21 C(=O)(C(CC(C)C)C(C)C)N1CCN(C(c2c(C)ncs2)=O)CC1C CCCCCCC(CC)NC(C1CCCN(C(c2cc(C)n(C)n2)=O)CC1)=O C1(CCOC)CCN(C(C2(CNC(=O)C(F)=CC3CC3)CC(C)(C)C2)=O)CC1 C1(C)(C(N2CC(CN(C(C(F)=C(C)C)=O)C)OCC2)=O)CCCCCC1 c1(C(N2CCCC(CC=C)(NC(C3CCC(F)C3)=O)C2)=O)c(C)cc(=O)oc1C CCC(C)C(O)C(=O)NCC1CC(NC(c2ccc(CO)nc2)=O)C1 C1(CCNC(CCN(CC(F)(F)F)C)=O)CCCCN1C(=O)C(F)C1CCCC1 C(=O)(C1=COCCO1)N1CC(C(C)NC(CC(C)CS(=O)(=O)NC(C)(C)C)=O)C1 C#Cc1cc(F)c(C(=O)NCC2CC(C)(C)CN2C(c2cc[nH]c2C)=O)cc1F C1(CC(C)NC(CC=C)=O)CC2CCC(C1)N2C(=O)Cc1ccc(C)cc1 c1(C(N(C2CN(C(CC(CC)CC)=O)CC2(C)C)C)=O)cnn2ncccc12 C(=O)(C(C)(C)C(=O)NCC1CC(O)CN1C(C1(N2CCCC2)CCCC1)=O)NC C1(C(N2CCC(SC)C2)=O)CC12CCN(C(=O)C1=COCC1)CC2 C(=O)(CC(C)(C)CC(F)F)N1CC2(OCC(NC(Cc3c(C)occ3)=O)C2)C1 CC1CC(C#N)(C(N2CCOC(CC(=O)NC(c3nncs3)C)C2)=O)C1 CC1(O)CCN(C(c2cc3c(s2)CCC3)C(=O)Nc2ccccc2)CC1(C)O C1(C(=O)NCC(=O)NCC(=O)NCC(CCC)C)CSCC(=O)N1 Cc1ccc(C(C)NS(=O)(=O)C2CC2c2cccc(F)c2)c(C)c1 Cc1nccc(Cl)c1C(=O)NCC1C(C)CCCN1C(=O)C1=NOCC1 C1(CNC(c2cn(CC=C)nn2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)CC1 c1(CNC(C)=O)ccc(C(=O)N(C2CC(NC(C3CC=CC3)=O)C2)C)cc1 Cn1cc(Cl)cc1C(=O)NC1C2CN(C(=O)CC3CNC(=O)O3)CC12 C1(NC(c2c(N)cccc2Cl)=O)CCN(C(=O)C(O)CC2CC2)CC12CCC2 C(=O)(C1=CCN(C(=O)C2=NOC(C)(C)C2)CC1)NC1C(CC)CCCC1 C1(C)(C(=O)NC(CCC)CNC(c2ccnc(O)c2)=O)CCC2CC2C1 c1(C(=O)NCCN(CCC)C(C2CC(C)CO2)=O)ccncc1-c1ccccc1 N1(C(c2cnn(C)n2)=O)CC(C(=O)NC2CC(=O)NC2=O)CCC1(C)C CC(C)CC(F)C(=O)NC(C)C(=O)NCCN(CCO)C(=O)OC(C)(C)C CC(C)(O)C(F)(F)C(=O)N1CCC(C(C)C(N2Cc3cccnc3C2)=O)CC1 N1(C(C(C)S)=O)CCc2[nH]nc(C(=O)Nc3ncc(Br)nc3I)c2C1 c1(NC2CCC(N)(CC(=O)OC)CC2)cccc(N=S(C)(C)=O)c1 C(=O)(CC(C)CC(C)(C)C)NCC#CC(N1CCCC(C)(CCC)C1)=O c1(N(CCCNS(CC)(=O)=O)C)ccc(C(F)(F)C(F)(F)F)cc1C c1(N(C)CC2C(C)C2)nc(=NCc2ccoc2)[nH]c2c1CSC2 C1(C(N(C(C)CCNC(c2cc(C(N)=O)c[nH]2)=O)C)=O)CN2CCC1CC2 C1(NC(C=C)=O)CCOCC1C(=O)Nc1cccc(OC(C)C)c1 CC1CC(CCNC(=O)C=C2CCC2)CCN1C(=O)CC(=O)NC1CC1 N1(C(c2c(C)ccc(O)c2)=O)CCCC(O)(CNC(=O)CN(C)CCO)CC1 C(CC(F)F)(C(=O)NCC1CC(C(C)(C)C)C1)N(C(c1ccc(C)nn1)=O)C c1(C(N2CCN(C(C3CC(=C)C3)=O)C3C2CC3)=O)cccc(C#CCO)c1 C(=O)(C1SCc2cccnc21)NC(C)CN(C(=O)COCC(F)F)C CC(C(=O)NCCCCNC(=O)C(c1ccccc1)Sc1ccnn1C)C(F)F N1(C(Cc2ccc(C)o2)=O)CCC=CC1C(N1CCC(N(C)C)CC1)=O C#Cc1cc(C(=O)N(C)CC2(O)CN(C(C3CCC3C)=O)C2)cc(Br)c1 N1(c2cc(C)ncn2)CC2CCN(Cc3cc4cc(Br)ccc4[nH]3)CC2C1 C1(CNC(CCN(CCCCC)C(C)C)=O)CC(F)CN1C(c1ccns1)=O C1(C(=O)NCCC(C)NC(c2cnc(C3CC3)nc2)=O)CCC(=O)N1C CCC(CCCC(=O)N1CCCC1C(C)(C)O)NC(c1cccc(=O)o1)=O CCC(C)CC(=O)C(=O)N1CC(C(O)C(N2CCC=CC2COC)=O)C1 CC1Cc2c(Cl)c(Br)cc(F)c2CN1N1CCCC1c1ncccn1 N1(C(CCC2C(C)=NNC2=O)=O)CCC(NC(=O)Cc2cc(C)on2)C12CCC2 N1(C(C2CCN(C(C(CC=C)C)=O)C2C(C)C)=O)CCC12CCC(C)CC2 C1(C(=O)Nc2c(CC)ccnc2)CC2(CCC2)CN1C(C1CCCC1C(C)C)=O CC1=C(C)CC(C(=O)NCC2C(C(=O)NC34CC3CN(C)C4)C2(C)C)CC1 N1(C(CCCC(C)C)=O)CCC(NC(c2csc(C(N)=O)n2)=O)C(C)(C)C1 CC(C)C(CC(=O)NC(C)CN(C)C(c1cnc(S)n1C1CC1)=O)C(C)C N1(C(c2nc(OC)oc2)=O)CCC2CN(C(C3CCC=CCCC3)=O)CC2CC1 C1(F)(CN(c2ncccn2)C(c2ccc(C3(O)COC3)cc2)=O)CCCNC1 C1(OC)CCN(C(=O)C(CC(C)C)ONC(c2n[nH]cc2C)=O)CC1F C(=O)(C1=CCC(NC(c2ccccc2F)=O)C1)NC(C1(O)CCC1)C C(CC(C)(C)C(=O)N(C)CC1CCCOC1)NC(C(n1c(C)ccn1)C)=O c1(NC(c2ccc(OC)c(Br)c2OC)=O)cc(C#N)c(F)cc1C CC(C)CCCC(C)C(=O)NCC1COCCN1C(c1ccnn1C)=O C1(C(N2CC(C(=O)NC(CN(C)C)CCO)(CC)C2)=O)CN(C)CCO1 C1(CNC(c2cc(C)[nH]n2)=O)CN(C(=O)CCCN2C(=O)CNC2=O)CCO1 C1(C)(C(=O)NC(CN(C(=O)Cc2sccc2C)CC)C)CCC2CC2C1 CCC(C(=O)N(CC(C)(C)CNC(c1ncccc1C(F)F)=O)CC)C(C)O N1(C(CCC)C(=O)NCCCC2CC2)CCc2c(O)cccc2C1 C(=O)(CC(C)C(C)(C)C)NCC(C(CC)NC(C(C(CC)C)=O)=O)(C)C C1(C(N(CCCCCNC(c2cn(CCC=C)nn2)=O)C)=O)CCC2(CC2)C1 C=CCC(C(=O)NC(CNC(=O)C=Cc1ccccc1)(CC)CC)OC Cc1ccc(C(=O)NC2(C3CN(C(C4(C#N)CC4)=O)C3)CC2)c(F)c1Cl N1(C(C(CCC=C)NC(=O)Cc2cccs2)=O)CC2C(=O)NC(=O)C2C1 c1(C(=O)NCCC(C)NC(CC=C=C)=O)cccnc1C(F)F c1(C(c2cccs2)NC(=O)NCCC(C)(C)O)ccc(F)cc1 C(=O)(CCCCCF)NC1C(OC)CN(C(=O)CCCC2CCOCC2)C1 N1(C(C(c2ccc(Cl)cc2)CC)=O)CCC(F)CC1(C)C CCC(C(=O)NCCCN(C(=O)C(C)COC1CCCC1)C1CC1)C(F)(F)F c1(C(=O)NC(C)CCNC(=O)CSc2nccn2C)sc(F)cc1Cl c1(CC)nc(C)[nH]c1C(=O)NC12CC(CNC(C3(O)CCOCC3)=O)(C1)C2 C1(N(C(CN(CC)CC)=O)CC)CCN(C(c2cc(C(F)(F)F)n[nH]2)=O)C1C CCC(C)C(C)C(=O)NCc1cc(C(=O)NCCC2(C)CC2)ccn1 C12(C(=O)NC3CC(OC(C)=O)C3)CCC(CN(C(C3(C)C=CCC3)=O)C1)C2 c1(C(=O)NC(CCOC)CNC(C2COCCOC2)=O)ccc(F)c(C)c1C C(=O)(C(CN(C)C)C(C)C)NC(COC)C(N1CCC(C(C)CO)CC1)=O C1(CNC(CC(C)N(C)C)=O)CCCN(C(=O)C(O)C2CCC2)C1 C(=O)(CS(=O)(=O)C(C)(C)C)NCC(c1ccccc1)NC(C1C(=C)C1)=O N1(C(c2cn[nH]c2)=O)CCC(F)(F)C(CNC(C2(F)CCCCCC2)=O)C1 N1(C(C2(C)CC(C)C2)=O)CC2(COC(CNC(=O)C(C)OCC3CC3)C2)C1 N1(c2cc(N(CC)CC3CCC(C)(F)CC3)nc(C)n2)CCCCC(S(C)(=O)=O)C1 N1(C(C2CCS(=O)CC2)=O)CC2CCC(C1)C2N1CCCCC1 C1(C(=O)OC)C2CC1N(C(C1(CNC(=O)OC(C)(C)C)CC(C)(C)C1)=O)C2 C#Cc1ccc(C(=O)NCC(O)CNC(=O)C(c2cccn2C)=O)cc1 CC(CCN(C)C)N=c1[nH]c(=NCC2(CN(C)C)CC2)[nH]c2c1CSC2 C1(C(=O)NCCn2c(CC)nnc2)CN(C(=O)C(C2(O)CCCC2)F)CC1C C1(C(=O)NCCN(C(C(CN(C)C)(F)F)=O)C)OCCOC12CCC2 CN1CCN(C(c2ccn(C)c(=O)c2)C(=O)NCCCC2CC2)CC1=O N1(C(C2C(C#C)C2)=O)CC2CN(C(C3(c4ccc(C(N)=O)cc4)CC3)=O)CC2C1 c1(C(=O)NCCC(C)NC(C2CC2(Cl)Cl)=O)cn(C)nc1-c1ccncc1 C(=O)(C(CCC1CCC1)NC(c1coc(CO)c1)=O)NC(C)Cc1nc[nH]n1 Cc1ncc(C)c(NC(N2CCN(c3ccccc3F)C(C)C2)=O)n1 C1(C(N(CC)Cc2ccc(O)cc2)=O)CCN(C(c2cc[n+]([O-])cc2)=O)CC1O N1(C(C(=O)N(C2C(=O)C2)CC(F)(F)F)=O)CC2CCCC(NC(=O)C(F)(F)F)C2C1 N1(C(C2CCC(OC)C2)=O)CC2=C(C1)CN(C(c1c(Br)cnn1C)=O)C2 C(=O)(C(CSC)NC(=O)C(F)CC1CCOC1)N(CC(=O)OC)CC1CC1 C(=O)(C(C)(C)C1CCN(C(=O)CC(C)O)C1)NCC(CO)OC c1(C(=O)NC2C(C)N(C(c3csc(O)n3)=O)CCC2)ccc2c(c1)CCCC2 CCC(CC)CC(=O)N1CCC1CC(=O)NC(C)(C)CCCOC C1(NC(=O)NCc2c(Cl)cn(C)n2)COc2ccc(F)cc2C1 N#Cc1nc(Br)cnc1NC(C1CCCN(C(c2cnc3snnc3c2)=O)C1)=O Cc1ccc(C(=O)NS(=O)(=O)CCN2CCCCC2)c(-c2ccccc2)c1 CC1CN(C(c2c(C(F)(F)F)ncn2O)=O)CCC1NC(C1CN(C(N)=O)C1)=O C1(C(=O)NC(C(CC)C)C(=O)OC)CCC2(CCNCC2)CC1 C(=O)(C(CC(C)C)NC(=O)OC)N(CC(CNC(c1noc(CC)c1C)=O)C)C Cn1c(C(N2CC(S)CC2Cn2cc(CCS(N)(=O)=O)nn2)=O)cc2sccc12 c1(C(N2CCC(CNC(=O)CC3COCCO3)CC2)=O)cc2cc(Cl)ccc2s1 N1(C(CC2(CNC(C3C(CCC)CCC3)=O)CC2)=O)CCC(C2(O)CC2)CC1 c1(NC(C)=O)cccc(F)c1C(=O)NC1CN(C(=O)C2CC2)CC1F C1(OCC)CCCN(C(=O)CN(C(=O)CCC(C)SC)C)C1 CC#CCCC(=O)N1CCCC(NC(C2CCC(N(C)C)CC2)=O)C1 C1(NC(C(C)Cc2ccnn2C)=O)COC2(C1)CN(C(=O)C#CC1(C)COC1)C2 N1(c2c(C#N)cncc2)C2CCC1CN(C(c1cc(CN)no1)=O)C2 C1(CNC(c2cn[nH]c2)=O)CN(C(c2cn(CC(F)(F)F)cn2)=O)CCCO1 c1(CC)csc(C(F)(F)C(=O)NC(CN2CCOCC2)CC)n1 Cc1cccc(OC(C)C(=O)NC(C)CC2CCN(C(C3CCC3)=O)CC2)c1 c1(CC)n[nH]cc1CN(C(c1cc(C(=O)OC)cs1)C(=O)NCCCSCC)C c1(OC)nccc(Br)c1C(N1CC(N(C2CCC2)C(C2C=CCCC2)=O)C1)=O N1(C(C(=O)NC2CCC(F)(F)CC2)CCC2CCCO2)CCC2C(C1)C2(F)F c1(CCC(=O)NCC(=C)CCNC(c2csc(O)n2)=O)ccncc1Br c1(C(N(C2CCC(NC(=O)Cc3ccon3)C2)C)=O)cc(C2CC2)ncn1 C12(CNC(C(C)=CC3CC3)=O)CCCC1N(C(=O)CC(O)C1CC1)CCC2 c1(CC(=O)NC2C(CNC(CN(C)CC)=O)CC2)c[nH]c2cc(Cl)ccc12 C1(C(C)C)CN(C(=O)CC2CCSCC2)CCN1C(C1CCOC1)=O CC1=C(C(=O)N2CCC(C)(NC(=O)CCC3CCCCN3C)C2)C(C)(C)CCC1 c1(C(=O)NC2CC(CNC(CC(COC)(C)C)=O)C2)ccc2c(c1)NC(=O)CC2 c1(C(=O)NCCNC(=O)C(F)(F)F)cnc2ccc(-c3c(O)cccc3F)cn12 c1(C(=O)OCC2(CC(=O)OC)CCOCC2)cc(Cl)c(Br)cn1 CN(C(=NCC12CC(CO1)C2)NCC1CCCCO1)Cc1cc(F)cc(F)c1 C=CCCCC(=O)NCC(C)NC(c1ncoc1-c1ccccc1F)=O c1(OC)cc(C(N2CCN(Cc3cnc(Cl)cn3)C3CC23)=O)cc(O)c1O C(N=c1nc2c(cnn2C)c(NCC2CC3CCC2CC3)[nH]1)c1ccc(SC)s1 C12(NC(=O)COCCOC)CC(NC(CC)CN(C(=O)CC(C)C)C)(CO1)C2 C1(N(C)C(c2ccc(C#N)s2)=O)CCCN(C(=O)CCNc2cncnc2)CC1 N1(C(CCSCCC)=O)CCN(C(=O)CC2CCN(C)C2)CC(O)C1 C1(NC(C2N(C(C)C)CCC2)=O)CC12CC(NC(=O)C1CC1)C2 N1(C(c2cc(CC)nc(O)c2)=O)CC2(COC(CNC(C3(F)CC3)=O)C2)C1 C(CC(C(=O)NCC[Si](C)(C)C)NC(=O)Cc1cnns1)OCC O=C1CC(CC(=O)N2CCC(O)(CNC(c3cncc(O)c3)=O)CC2)=NN1 N1(C(C(CCC)OCC)=O)CCC2(CC1)OCCC2NC(c1cnccc1Cl)=O c1(OC)cc(C)c(C(=O)NC2(CNC(=O)CC(C)CF)CCCC2)cn1 C1(C(=O)NC(C(C)C)(C)C)CCN(C(=O)CCn2ccnc2)CC1 N1(C(c2c(C)nsc2)=O)CCC2(C1)CN(C(=O)CCC1CC1)C2 c1(N2CC(=C(CNC(c3cnc(C)[nH]3)=O)F)C2)cncc(Cl)n1 N1(C(CC)=O)CCCC(O)(CNC(c2cccn(C3CCSC3)c2=O)=O)CC1 N1(C(c2cc(OC)nc(Cl)c2)=O)CCN(C(=O)CC(C)N(C)C)C2CCC12 C1(CC(=O)N(CC(C)NC(CCc2onc(C(C)C)n2)=O)C)CCCC1(F)F C(=O)(C1CCCc2cncn21)N1CCC(COC)(NC(c2cc(CO)[nH]n2)=O)C1 N(S(=O)(=O)N1CCCC1C)C(CCC)Cc1ccc(C(F)(F)F)cc1F N1(C(C(CC)COC)=O)CCC2C(NC(c3ccccc3SCCO)=O)CC12 N1(CC(=O)NCCc2ccn(-c3ccccc3)n2)CCCCC1Cn1ccnc1 Cc1cccc(C)c1C(N1CCN(C(c2ccc3c(c2)CC3)=O)C(C)C1)=O C1(C(=O)NCC2C(NC(C(C(=O)OC)(C)F)=O)CC2)CC2(C1)CC(F)(F)C2 C(=O)(CCCC(=O)N(C1CCN(C(=O)C(CSC)OC)CC1)C)N(CC)CC C1(CNC(c2nc(COC)sc2)=O)CC2(CC2)CN1C(=O)C(C)n1cccc1 CC1SCCCC1C(=O)NC1(C)CC(C(=O)NCCOC2CC2(F)F)C1 C(C1CCCCCC1)=CC(=O)NC(CC(C)C)CNC(=O)CC1CCC(C)(C)C1 CCS(=O)CC(=O)NCCC1(CNC(c2[nH]ccc2-c2cccs2)=O)CC1 C1(C(N2CCCC(OC)C2)=O)COC2(CCN(C(c3cc(Br)cnc3F)=O)CC2)C1 N1(C(C2(CC=C)CC2)=O)CCCC1CNC(=O)C(O)CC1CC1 CC(C)(O)C(F)C(=O)N1CCC1C1CCN(C(c2ccn(CCF)n2)=O)CC1 c1(OC)cnccc1C(=O)NC(C)C(C)NC(=O)C(F)(F)c1csc(=N)[nH]1 C(C(C)(C)CC(=O)Nc1cncnc1C)NC(c1oc(CC)c(C)c1)=O C1(NC(C(CC)C)=O)C2CC3C1C3C2C(=O)NC(C1CC1C(=O)NC)C c1(C(=O)NC2CCC(NC(C3C(F)(F)C34CCC4)=O)CC2)c(F)ccc(F)c1F N1(C(c2c(C)n(CCO)nc2)=O)CC2CCC(N(C(=O)CC(C)F)C)C2C1 S(=O)(=O)(c1ccc2oc(O)nc2c1)N1CCC(F)(C(N2CC(O)C2)=O)CC1 c1(C(=O)OC)nccnc1CNC(=O)N(c1ccc(Cl)cc1)C.c12ccccc1O2 c1(C(=O)NCC(CN(C(c2cccc(C3CC3)n2)=O)CC)(C)C)cc[nH]c(=N)c1 CCCCC(O)C(=O)NCC1CC2(CC2)CN1C(C1CCCN(CC)C1)=O N1(C(c2nc(C)oc2)=O)CCOC2(CCCN(C(c3c(C)nsc3Cl)=O)C2)C1 c1(C(=O)NC2CN(C(C3ON=C(C(C)C)C3)=O)CC3C2C3)ccc2c(cnn2C)c1 C(C(C)C(F)C(=O)NC(CCO)C(F)(F)F)NC(C1C(C(=O)OC)C=C1)=O c1(C(N2C(C)CC(NC(c3cc(C)sc3)=O)C2)=O)nc(OC2CC2)ccc1Cl CCS(=O)(=O)CC(=O)NC(C1CCCN1C(=O)Cc1ccccc1C(C)C)C c1(CC(=O)NCC2(OC)CN(C(c3cncc(C)c3)=O)C2)ccccc1SC C(=O)(C1CCc2snnc21)NC1CCCC(NC(C(C)(C)n2ccnn2)=O)C1 N1(C(=O)CNc2nnc(-c3ccccc3)s2)CCC(C(F)(F)F)C(F)(F)C1 C1(NC(C2(CCC=C)CN(C(C3CCCC3O)=O)C2)=O)CC=C(C)CC1 Cc1ccc(C(=O)NCC2(C)CCCN2C(C2COC(C)C2)=O)cc1N C(N=c1nc2ncn(C)c2c[nH]1)C1CC(C)N(Cc2ccccc2)C1 N1(Cc2nc(-c3ccc(OC)cc3)oc2)CCC2(CC1)CNC2C(C)C c1(CC(=O)NCCC2(O)CN(C(CC(CC)O)=O)C2)c(F)cc(F)cc1F c1(CC(=O)NCC(CCCC)NC(C2CC2COC)=O)noc2ccccc12 C1(CNC(=O)C(O)c2ccsc2)CCN(C(=O)CC2CCCCO2)CC1 C1(C(=O)NCCN(CCC)C(c2cc(CC)nnc2C)=O)CCn2ccnc2C1 c1(C(=O)NCC2(CC3CC3)CN(C(CN(CCC)C)=O)C2)ccncc1C(N)=O C(=O)(C(O)CC(N)=O)NCCCN(CCCNC(CN(CCC)C)=O)C C(=O)(C(C)CC(F)(F)F)N1C(C(=O)NCC2(C#C)CCC2)COCC1 S(=O)(=O)(c1cc(C(=O)NC(c2ccncc2)(C)C)ccc1Cl)NC(C)(C)C C(C(CO)(CO)NC(c1cc(C2CC2)nn1C)=O)N(C(=O)CC1CCCC1)C c1(C(N2CCC(CNC(c3ccccc3C(F)F)=O)C2)=O)c[nH]c(=O)cn1 C1(CNC(CC2CC(C)(C)OC2)=O)CC2(CC2)CN1C(C1CCCC(F)(F)C1)=O C1(C)(C(=O)OCC)CC(C(N2CCCC2C(C)NC(=O)C(C)OC)=O)C1 N(C1CCc2ccc(Cl)nc21)C(C(C)NCc1nc[nH]n1)=O C(=O)(C(CC)C(C)(C)CC)NCC(CC)NC(c1ccnc2c1ncn2C)=O C1(CCNC(CCc2onc(CC)n2)=O)CN(C(=O)C(F)=CC2CC2)CCO1 c1(C(=O)NC2CN(C(C3(Cl)CC3)=O)CC2C2CC2)cc(=O)n2ccsc2n1 Cc1nc(C(=O)NCCC(O)CNC(=O)C=CC2CCC2)cc(O)n1 N1(c2cc(C)ncn2)CCC(O)C(C(=O)NCCOCc2ccccc2)C1 c1(C(N2C(CCC(=O)NCCn3ncnn3)CCC2)=O)cc(=O)cc[nH]1 C(C)(C)(C(=O)NCC1CCN1C(=O)Cc1csc(C(=O)OC)c1)OCCC N1(C(COC(CC)(C)C)=O)CC(C)CN(C(=O)CCCc2ncco2)CC1C C12(NC(C(=O)NC(C)C)=O)CCCN(C(C3CC(=O)N(C)C(=O)C3)=O)CC1C2 N1(C(CC(C=C)C)=O)CCN(C(=O)C(CC)(CC)CO)CC2(CC2)C1 C1(NC(c2ccccc2Cl)=O)(CO)CCN(C(=O)CCC(F)(F)F)CC1 N1(c2snc(COC)n2)CC2CC1CCC2NC(C1CCc2nn[nH]c2C1)=O N1(C(Cc2c(C)sc(Br)n2)=O)CC(C)c2ccccc21 Cc1cc(CC(=O)NCCC(C)NC(=O)Cc2ccco2)on1 C12(NC(CCC(=O)NCC)=O)CCCCCC1N(C(c1cccnc1F)=O)CC2 N1(C(c2cc(C)on2)=O)C2CCC1CC(F)(CNC(=O)C=CC(F)(F)F)C2 CCCC(CC(C)C)C(=O)NCCC(C)(C)NC(C1COC2(CCC2)C1)=O CC(C)(C)CC(O)C(=O)N1CC(C2CC2)(C(N2CCS(=N)(=O)CC2)=O)C1 CC1CN(C(=O)CC2CC3(C2)CN(C(=O)CCCCN=[N+]=[N-])C3)Cc2c[nH]nc21 c1(CC(=O)NC2C(C)N(C(C3CC3F)=O)CC2)cc2ccccc2cc1O c1(C(N2C3CC(NC(C(C(C)C)SC)=O)C3CC2)=O)ccc(Cl)c(Cl)c1O N1(C(c2cc(C)c(=O)n(C)c2)=O)CCC2(CC1)CN(C(C1CC1C)=O)CC(C)O2 Cc1n[nH]c(C)c1CCNC(C1CSCN1C(=O)CCCn1cccn1)=O CCS(=O)(=O)CCNC(=O)C=CC(C)(C)NC(=O)C=CCNC(=O)CC(C)(C)C N1(C(=O)CSc2n[nH]c(O)n2)CCCN(C(c2cccc(F)c2F)=O)CC1 N1(C(CP(C)(C)=O)=O)CC2CC(NC(C3(F)CCCCC3)=O)CC1C2 N1(C(CCSCCC)=O)CCC(C)(CNC(=O)C(C2CCC2)OCC)C1 C1(NC(CCN(C)CC2CCCCC2)=O)CC(C(=O)NOCCO)=NO1 N1(C(C(CC)=CC)=O)CC(C)CN(C(=O)C(C)(C)N(C)C)CC1C N1(C(C(=CC2CCCC2)C)=O)CCN(C(C2CCS(=O)(=O)N2)=O)C(C(C)C)C1 C1(NC(Cn2c(C)cc(C(F)F)n2)=O)CC2CC1N(C(C1C(C)C1C)=O)C2 C1(C(N2CCN(C(c3n(C)cc(Cl)c3)=O)C3(C2)CC3)=O)COc2ccccc2O1 C1(CNC(CSC(C)C)=O)(CO)CCCN1C(C1CC(CN(C)C)C1)=O N1(C(C(C)(O)C2CC2)=O)Cc2ccc(CNC(c3ccn(C(F)F)n3)=O)cc2C1 C(=O)(C(CO)NC(=O)Cc1ccon1)NC1(C(N)=O)CC1 c1(C(N2CCC(N(C)C(=O)OC(C)(C)C)C2)=O)cncc2nc(O)[nH]c12 CC12CC(C(=O)NCCC3CCC4(CC3)CC4)(C1)C1(COC1)O2 O=S(=O)(c1cncc(Br)c1Cl)NCCCc1ncc(C(=O)O)[nH]1 CCCC(C(=O)N1CC(NC(=O)C(OC)OC)C(CC)C1)NC(=O)OC Cc1ccc2c(c1)CCN(C(C1CC(=O)N1)=O)C2 C(=O)(C1=CCCC1(C)C)NCCCN(CCCNC(c1cnc(C(N)=O)s1)=O)C C(=O)(CCCC(=O)NCc1ncoc1C1CCN1C(=O)COC1CCCCC1)OC O=C1CSc2ncc(C(=O)NC3CC3CNC(C3(Cl)CC3(F)F)=O)cc2N1 C(CC(C(C)C)NC(c1cn(CCOCC)nn1)=O)NC(C1C(=C)CC1)=O c1(CC)ccc(N)c(C(N2CCCC2C(C)NC(=O)C(F)(F)CO)=O)c1 c1(C(N2CCN(C(c3cc(C)ncn3)=O)C(CO)C2)=O)c([N+](=O)[O-])c(C)nn1C Cc1cc(C(=O)NC2(CO)CCCN(C(c3snnc3C)=O)C2)cc(Cl)c1 c1(C(=O)NC2CCN(C(C3(N(C)C)CC3)=O)C2)cc(O)ncc1Br c1(C(N(CCNC(C(C(C=C)C)C)=O)CC2CC2)=O)cccc2cnnc(O)c12 CC(C(O)C(F)F)NC(c1cnn(CCNC(=O)CCc2cnn[nH]2)c1)=O N1(C(c2c(CC)nc[nH]2)=O)CCCN(C(=O)CCC(C)(C)C)C(C)C1 Cc1ncc(Cl)c(C(N2CC(NC(c3cc[nH]c3)=O)CCC2C)=O)n1 C=CC(CC)CC(=O)NC(C(=O)Nc1cnc(CO)nc1C)C1CC1 c1(OCC)ccc(C(C)NC(=O)NCCNS(N)(=O)=O)cc1.C1CCC1 C(CC(O)C(=O)N1CC(N(C)C(C2(C(F)(F)F)CCCCC2)=O)C1)OCC c1(C(N2CCC(C)(NC(c3ncn(C)c3)=O)C2)=O)cc2cccc(Cl)c2s1 n1(CC)ncc2cc(C(=O)NCCC(C)CCNC(=O)Cc3ccco3)cnc12 Cn1ncc(CNC(c2nc(Cl)cs2)=O)c1C(=O)NC1CC(CC(F)F)C1 c1(C(=O)NCC2CC(NC(=O)COc3ccc(F)cc3)C2)ccccc1[N+](=O)[O-] c1(C(N2CC(C(N)=O)C(NC(=O)C(F)C3CCC3)CC2)=O)ccn2c1CSCC2 C1(N(CCN(C(C)(C)C)C)C(=O)C2CC2)CCN(C(=O)C(N)=O)CC1 c1(NC(C2CCCN(CC3CC3)C2)=O)c(OCC2CC2)cccc1Cl N1(C(Cc2c(Cl)cn(C)n2)=O)CCC(NC(=O)CCN2CCCCC2)C(CO)C1 S(=O)(=O)(CC(=O)NC1CC(N(C)C(c2ccc(C3CC3)s2)=O)C1)NC N1(C(=O)NCC2CCCO2)CCC(c2nc(=O)o[nH]2)CC1 n1(CC(=O)NC(CCNC(C=C(CC)C)=O)C)sc2ccccc2c1=O C1(C(=O)NC(CN(C)C)C(N2CCC(O)(CN(C)C)C2)=O)Cc2nccn2C1 Cn1ccn2ncc(C(N3CC4(CC(NC(c5ncc(Cl)n5C)=O)CO4)C3)=O)c12 C1(NC(c2c(N)ccc(OC)c2)=O)CN(C(=O)C(C)C(C)O)CC12CCOCC2 C1(OC)CC2CC1CC2(C(C)C)OCc1cn(C2(C(=O)OC)CCOCC2)nn1 c1(C(=O)NCC2(CNC(C(C3CC3)OC)=O)CC2)cc(C(C)=O)on1 N1(C(c2ccccc2CO)=O)CC2CC1CN2Cc1ccncc1Br C1(C)(NC(C(CCSC)NC(c2nc(Cl)cs2)=O)=O)CC(C)(C)OC1=O C12(C(N3CC=CC3CO)=O)CCC(=O)C1CNC2 C(=O)(CC1=CCCCC1)NC(C(CO)NC(C(c1c(C)nn(C)c1C)=O)=O)C c1(CNC2CCC(C(=O)Nc3cccc(CC)n3)CC2)cccc(C)c1F c1(OCC(c2n(C)ncc2)(c2nnnn2C)NC2CCCCO2)cccc(Cl)c1 C(C(CN=c1[nH]c(=NCCC(C)OC)[nH]c2c1CSC2)OC)OC Cc1cc(C(=O)NCC2(O)CC(NC(=O)C(F)Cc3ccccc3)C2)no1 c1(C(=O)NC2CC(C)(NC(CC(C)(C)OC)=O)C2)[nH]cc2c1CCS2(=O)=O c1(C(=O)NC(C)CNC(C2(C(F)(F)F)CC=CCO2)=O)cnc2ccccc2c1 c1(C(N2C(C)CN(C(C3CCS3(=O)=O)=O)CC2)=O)nccc2ncncc12 C(=O)(C1CCc2ccccc21)N1CCC(CC=C)(NC(=O)C(C)=CCC)C1 n1(C(C(N2CCC3C(NC(CC(C)C)=O)C32)=O)C)c(=O)oc2ccccc12 C(=O)(CCCC(F)(F)F)N1C(C)CC(CNC(C2COC(=O)N2C)=O)C1 C(=O)(CCCN=[N+]=[N-])N1CC(CC(=O)N(CC(C)SC)C)OCC1 C(=O)(CS(=O)(=O)CC)NC(CCCC)CNC(C1C2CCC1CC2)=O O=C1NC2CN(C(C3CC(O)CN3C(C3CCCOCC3)=O)=O)CC2O1 C12(CNC(c3cnc(OC)s3)=O)CCC(CC1)N2C(=O)Cn1ccnn1 N1(C(c2c(C)c[nH]c2)=O)CCC2(C=C(C(=O)NCC(C)(O)CC(C)C)C2)C1 Cc1cccc2c1CC(C(=O)NC1CCC(NC(C3CC3C)=O)CC1)O2 O=S1(=O)CC2CN(Cc3ccc(I)c(F)c3)CC2C1 c1(C(=O)NCC=C(C(=O)N(C(CC)C2CC2)C)C)nccnc1N CC(CC1=CCCCC1)NC(c1cn2c(n1)CCCC2)C c12ccc(cc1)OC2.c1(OC)ccsc1CNC(c1nnnn1C)COC N1(CCN(C(CC2(NC(C3C(C)(CC)C3)=O)CC2)=O)C)CCOCC1 c1(C(=O)NCC(CC)NC(=O)CC2(c3ccccc3)CC2)cnccc1N(C)C N1(C(C2C(C)CC(C)O2)=O)CC=C(CNC(=O)C(N)=O)CC1 c1(C(=O)NC2C3CCN(C(C4CC5(CC5)CO4)=O)C23)cc(Cl)c(Cl)c(Cl)c1 CCC(C(=O)NCC(=O)NCC1CCN(Cc2ccccc2)CC1)C(C)O C(CCCC(=O)NC1(C2CCCN2C(=O)CCC2CCCO2)CC1)N(C)C N1(C(CCC)=O)CC2(C1)CN(C(=O)C(c1ccccn1)O)C2 CC1(C(N2CCC2C(=O)NCC2=CCCOC2)=O)CCNC1=O N1(C(C)=O)CCCC(C(N2CCC(N(C)C(C3CC4(C3)CC4F)=O)CC2)=O)C1 c1(C(N2CC(CC)(CNC(C3CN(CC)CCO3)=O)C2)=O)cc2n(n1)CCC2 c1(NC(COCC)=O)ccc2c(c1)CCN(C(C)(C)C)C2.c12ccsc1C(=O)N2 c1(C(C2(C3CC3)CC2)N(C)C)cccc(OCC(=O)N(C)C)c1.C(C)(C)(C)ON N1(C(CCCSC)=O)CC2C3CCC(C2C1)N(C(c1cc(C)n(C)c1)=O)C3 c1(C(=O)NC(CCNC(C2C(C)CC2C)=O)(C)C)cc(Br)c(CC2CC2)s1 c1(C(=O)NC(COC)C)cc(-c2ccc(O)c([N+](=O)[O-])c2)nc2ccccc12 c1(OC)ccnc(C(N2CC(N(C(=O)C(F)=CC3CC3)C)C2)=O)c1 O=C(C1Cc2ccccc21)N1CCCC(CNC(C23CCC(CC2)O3)=O)C1 c1(NCc2cn(CCC(=O)NCC3CC(F)(F)C3)nn2)c(F)ccc(Cl)c1F c1(C(N2CCC(O)(CNC(=O)CCC(F)F)C2)=O)cc2ccc(F)cc2[nH]1 N1(C(c2ccn(C)n2)=O)CCCC(C(C)(C)C(=O)NCc2ccncc2F)CC1 N1(C(C2C(C)(C)C2CNC(=O)C(C)(C)n2cnnn2)=O)CCCC(F)CC1 C=C(C)C1OCCCC1C(=O)NCC1=CCCN(C(=O)Cc2cncs2)C1 CC(C)C(F)C(=O)NCCN(C(C1CCC1C)=O)Cc1ccc(Cl)nc1 c1(C(N(CCNC(C2(CC)CN(C(C)=O)C2)=O)CC)=O)nn(C(C)(C)C)cc1Cl C=CCC(CC(F)F)NC(=O)CC1CCCN(C(=O)Cn2cc(CO)nn2)C1 CC1CN(C(=O)CC2OCCO2)CCC1CNC(C1CC(O)C1)=O C1(NC(CSC)=O)CC(C)CN(C(C23CC(F)(C2)C3)=O)C1 c1(C2(C(=O)NCC(C)(C3CC3)NC(CC=C)=O)CC2)cc(F)cc(C#N)c1 c1(C(=O)NCC(C)N(C(CCCc2ncc(C)o2)=O)C)cc2ncccn2n1 N1(C(C2(C=C)CCCC2)=O)CC(C(=O)Nc2cnn3ccccc23)C2(CCC2)C1 C1(C(=O)Nc2ccc(C)nc2I)CC12CCN(C(c1c(Cl)cncc1Cl)=O)CC2 C(=O)(C(C)CC(F)(F)F)N1C2CC(NC(c3c(C)nc(Br)o3)=O)C2CC1 c1(CC(N2C(CC(=O)N(c3ccccc3)CC)CCC2)=O)ccc(F)c(Cl)c1F N1(C(C2(SCC)CC2)=O)CCC(C)C(NC(=O)C(C)=O)C1 c1(CN2C(CNC(CC(C)C)=O)CCC2)cccc2c1oc1ccccc21 c1(C(=O)NCC(CO)NC(=O)C2=CCOCC2)nnc(O)c2ccccc12 C(=O)(CC(C)N(C)C(c1c[nH]nc1CNC(c1cc(C)no1)=O)=O)OC c1(C(C(=O)NC2CC(NC(C=C(CC)CC)=O)C2)=O)ccc(O)cc1 CCC(CC)C(F)C(=O)N(CC(O)CNC(=O)CC(CC)C1CCC1)C c1(C(=O)NCCNC(C2CC2)=O)ccc2nccn2n1.O=C1CCN1CCC C1(COC)(NC(=O)Cn2cc(C)cn2)CN(C(C2CCN(C(C)=O)C2)=O)C1 N1(C(c2ccn(COC)n2)=O)CCC(C2CC2)(NC(c2cn(C(C)C)nn2)=O)C1 c1(C(=O)NC(C)(C)C(O)C(F)(F)F)cccc(S(=N)(=O)C(F)F)c1 c1(OC)cccc(N2CCC(C(=O)N(C(C)C(=O)O)Cc3ccccc3)C2)c1 c1(C(N2CCC(N(C(CCC=C=C)=O)CCO)C2)=O)cnc2c(cnn2C)c1 Cc1c(O)ccc(C(=O)NC(CNC(=O)C(CC2CC2)CC2CC2)CO)c1C Nc1c(Cl)cc(NC(C2CN(Cc3cccnc3F)CC(F)(F)C2)=O)cc1Cl CON(C(=O)C=CCNC(c1cc2ccccc2o1)=O)C(C)C c1(C(=O)NC2(C)CCN(C(C3CCC3C(F)(F)F)=O)C2)cccc2c[nH]nc12 N1(c2c(C)cncn2)CCC(O)(CC(=O)N(C)CCN(C)C)CC1 N1(C(C(C)OCCC(C)C)=O)CC=CC1CNC(=O)Cc1ccon1 C1(C)(OC)CC2CC1CC2NC(=NCc1cnccc1Cl)NC1CCCCC1 c1(C(=O)NCCN(CC(C)O)C(c2n(CC)ccc2)=O)cnc(N(C)C)cn1 C1(NC(c2cc(C)oc2)=O)C(C)CCN(C(C2CCCSS2)=O)C1C CC1(C(=O)NC2CCN(CCNC(C3CCCCNC3=O)=O)CC2)CCC2CC2C1 C(CC1=CCN(C(C2(NC(C)C)CCC2)=O)CC1)NC(Cc1c(C)cco1)=O c1(CNC(C(CC)C(C)O)=O)ccc2c(c1)CCCC2NC(c1cc(C)[nH]n1)=O N1(C(CC=CCC)=O)CCCN(C(=O)C(=O)Nc2ccccc2)C(CO)C1 C(C(=O)NCC(C)NC(c1nccc(C(F)F)n1)=O)(C(C)C)SCC c1(C(=O)NCC(CCCC)NC(=O)CCOC(C)C)[nH]cc2c1CCC2 N1(Cc2cc(NC(c3c(C)cc(Br)nc3)=O)ncc2)CC2CC1CS(=O)(=O)C2 CCC(C(=O)N1CCC1CNC(c1cc(S(C)(=O)=O)oc1C)=O)C(C)(C)CC c1(NC(C(C)(F)F)=O)cccc(NC(=O)CCc2cncnc2O)c1 C(C(CC(C)C)C(=O)N1CC(C(N)=O)(CNC(=O)C=CC2CCCCC2)C1)OC Cc1ccn(C)c1C(N1CC=CC1CNC(C1(c2ccc(F)cc2)CC1)=O)=O C=CCC(CC(F)F)C(=O)NC1C=CCN(C(C2OCCOC2C)=O)C1 CC(CNC(=O)C=Cc1ccoc1)CC(=O)NCC(O)Cn1cccn1 C(=O)(C(CN=[N+]=[N-])NC(=O)Cn1cncn1)N(CC(N1CCCC1)C)C C(=O)(CC(F)(F)C(F)F)N1C(CCC)CN(C(c2cn(C(C)C)cn2)=O)CC1 S(=O)(=O)(c1cccc(=NCCCCCCF)[nH]1)NC(C)C(C)S(C)(=O)=O C#CC1CN(c2nc(C3CC3)nc(C)c2Br)CCN1C C(=O)(C1OCCn2ccnc21)NC12CN(C(c3scc(C)c3C)=O)C(CC1)CC2 c1(C(=O)NC(CCN(C(COCCCCC)=O)C)C)ccc(OC(F)F)cn1 CC1(C)CC(CC(=O)NOCc2ccccn2)N(C(=O)CC2CC=CC2)C1 c1(OCC(=O)NC2CC(CNC(C3(C)CC3(Cl)Cl)=O)C2)cc(Cl)cc(Cl)c1 c1(OC(COC)C(=O)N2CCC(c3ccc(Cl)cc3)C2)cc(F)cc(F)c1 N1(C(c2c(C(=O)O)c(Br)ccc2)=O)CCC2(CC1)CC(c1ccc(Cl)cc1)C2 c1(C(=O)NCC(CC=C)NC(=O)C=CC=CC)c(C)cc(C)cc1N C1(OC)(CNC(=O)COC2CC2)CCN(C(c2cccc(C(C)(C)C)c2)=O)CC1 Cc1cnc(C(=O)NCCCN(C)C(C2CC2c2ccsc2)=O)cn1 N1(C(c2c(Cl)ccc(C#N)c2)=O)CCC2CN(C(=O)CSC(F)(F)F)CC2C1 c1(C(n2cc(COC3CCNCC3)nn2)CN)ccc(F)cc1 Cc1ccc(O)nc1CNC(C1(NC(C2CCC(=O)C2)=O)CC(CO)C1)=O C(=O)(C(CC(F)F)SC)NC1(COC)CN(C(=O)CC2OCCCC2(C)C)C1 C(=O)(CC(C)(C)CC(F)F)NCC1CCN(C(c2c(OC)ccs2)=O)CC1O Cc1nn(CC(N2CC(NC(C3(C)CC(F)C3)=O)CC(F)C2)=O)c(C)c1C=NO N1(C(C(C)=CC2CC2)=O)CCCC(O)(CNC(=O)Cn2cnc(C(N)=O)n2)C1 C(CCCCCNC(=O)Cn1c(C)csc1=O)NC(CSc1nc(C)[nH]n1)=O c1(CC(=O)NC2C(C)N(C(c3cnn[nH]3)=O)CC2)ccc(Br)c(F)c1 c1(C(=O)NCCCN(C(=O)C(F)C2CCOC2)C2CCCC2)cc(C2CC2)on1 c1(C(N2CCCCC(CNC(C3CCC(O)C3)=O)C2)=O)ccc2c(n1)NCCO2 N1(C(C(CC)N(CC)CC)=O)CCC(COC)(NC(c2sc(=N)[nH]c2C)=O)C1 C1(NC(=O)CC=C(Cl)Cl)CCN(C(=O)COCCc2ccccc2)CCC1CO N1(C(C2C(CC)CCO2)=O)CCCC2CN(C(=O)CN3CCC(C)CC3)CC12 C(C(C)C(=O)N(CCO)OC)N(C(CC(CC)CC)=O)C C(=O)(CC(F)(F)CC(=O)NC1CN(C(c2c(C)n[nH]c2C)=O)CC1C)OC CC1=C(C(=O)NC2CCC(CNC(c3cc(O)ccc3O)=O)C2)SCCO1 N1(C(=O)COC)C2CCCC1CC2.C12CCN(CC1)CCN2C(=O)SC(C)(C)C C(=O)(CC(C)C(C)C(C)C)N1CC(C2(NC(c3onc(C)c3C)=O)CC2)C1 C1(C(N(C(CNC(Cc2cccc(SC)c2)=O)C)C)=O)CCOC2(CCCC2)C1 CCCC(C)CC(=O)NC1(CC(=O)Nc2cc(CO)cc(F)c2)CC1 N1(C(c2cnc(OC)c(C)c2)=O)CCCCCC(NC(c2scnc2C)=O)C1 c1(OC)ccc2[nH]c(C)c(C(=O)NC(CNC(=O)C=CSC)C(C)(C)C)c2c1 C1(C(CNC(CN(C(C)C)C)=O)F)CCN(C(=O)CC(F)(F)F)CC1 c1(NC(CC(C)C2CCCO2)=O)cncc([N+](=O)[O-])c1 c12ccc(nc1)S(=O)(=O)NCC(OC)CNC2=O.C1(COC)(CO)CCCC1 N1(C(C2(C)CC2Br)=O)CCC2(CC(NC(=O)COc3ccccc3F)C2)C1 C1(NC(=O)NCc2onc(C(C)OC)n2)CC2(CCCO2)C1 C1(CC=C)(NC(c2cc(C)c(Br)s2)=O)CCN(C(=O)C=CC)C1 C1(CCNC(C2(OC)CCC2)=O)CN(C(=O)OC(C)(C)C)CC1C C(CCC(C)C)(C(=O)N1CCCN(C)CC1C)NC(CC1(CC)CCC1)=O C(=O)(C(C)CC(F)(F)F)N1C(C(=O)NC2CN(CCC)C2)CC(=O)C1 N1(C(C2(SC)CCCC2)=O)CCC(O)(C(C)NC(=O)COCc2scnc2C)C1 Cc1sc(Br)nc1C(=O)NC1CCCC1CNC(=O)C(C)CC1CC1 c1(C(C(=O)NC(CC#C)COC)C)ccc(C(F)F)cc1 C(CCCC(=O)N(C(C)CCNC(=O)CC1(CO)CCOCC1)C)OCC Cc1n[nH]c(C)c1CCC(=O)NCC(C1CC1)N(C(=O)CC1CCC(C)O1)C N1(C(CCC(=O)OC)=O)CC2CC(NC(c3c[nH]cc(C)c3=O)=O)CC1C2 CC(C)(C)C(O)C(=O)NC1(C)CN(C(=O)Cn2cnc(Br)c2)C1 C1(NC(CC)=O)C2CC(NC(=O)C(C3(O)CCCC3)F)CC12 C(=O)(C(F)(F)F)NC1CCN(C(CSCC(=O)Nc2ncccn2)=O)C1 C(CC(C)CC)(C(=O)NC1CN(C)CCC1O)NC(C(CC=C)CC)=O N1(C(Cc2c(C)cccn2)=O)CC(CNC(=O)C(F)(F)C2CCCC2)C(C)(C)C1 c1(C(N2C3C(NC(=O)CC4CC=CCC4)CC(C3)C2)=O)c[nH]c2ccc(Cl)cc12 c1(CN(C(=O)CC2(C)CC2(F)Cl)C)cnn2c1CN(C(=O)CC1(O)CCC1)CC2 CC12CCC1CN(C(C1CNCC13CCC3)=O)C2 N=c1[nH]c(Cl)c(Cl)c(=NC2CCCC(CO)C2)[nH]1 c1(C(=O)NCC2CCC2NC(C2CC2(F)F)=O)cc(C2CCCCC2)on1 CON=C(C(=O)N1CC(=C(F)CNC(=O)CCCN=[N+]=[N-])C1)c1ccco1 N1(C(C=CSC)=O)CC2CC(NC(=O)Cc3ccc(F)cc3)C1C2 c1(C(=O)NCC(CNC(CCC(=C)C)=O)C)cccc(Cl)c1C N1(C(CCC)=O)CCCC2(CCN(C(=O)CC3(O)CCCOC3)CC2)C1 c1(C(N(CC(C)NC(C2CCCC(C(N)=O)C2)=O)C)=O)ccc2[nH]ccc2n1 c1(C(=O)NC(C2CCCCC2)C(=O)N(C2CCCC2)CCO)cccc(CO)n1 CCCCCCCCc1ccsc1C(=O)NCC(O)CNC(c1cc(Cl)c[nH]1)=O CC1=NS(=O)(=O)N(C)C=C1C(=O)NCC1(NC(=O)C(CC(C)C)NC(N)=O)CC1 N1(C(C(C)C(C)(C)C)=O)CC(NC(c2cnn(C)n2)=O)CC12CCC2 CC1(C)CN(C(C23CCCC2C3(F)F)=O)CC(C)(C)C1NC(=O)Cc1cccs1 c1(Cn2cc(C(C)(C)OC)nn2)ccc(-c2ccc(Br)cc2)cc1 N1(C(C(C)SC(F)(F)F)=O)CC=CC(NC(=O)CCc2ccccn2)C1 c1(CC)c(C(N2CCN(C)C(CNC(=O)C(C)(CC)CO)C2)=O)cccc1C c1(C(=O)NCC2CN(C(=O)C(O)C3CC3)CC2C(F)(F)F)ncc(Cl)cc1F C12(NC(C(C(C)C)C)=O)CCCC1N(C(C1CCCCN(C)C1=O)=O)CCC2 CCC(C)CC(=O)NC1CC(c2ccccc2)(NC(=O)CC2CNC(=O)C2)C1 N1(C(c2c(CNC(CN(C3CC3)CC)=O)ocn2)=O)CCNC(=O)CC1 C1(C)C(=O)N1.c1(CN(CCN(C(C2(C(C)OC)CC2)=O)C)C)cocn1 c1(CC)c(C(N2CCC2C(=O)NCc2ccccc2OCCO)=O)cnn1CC C1(O)(C(C)NC(C2C(CC)C2)=O)CCN(C(C2CCCOC2)=O)CC1 N1(C(C(CC)CC)=O)CCCC(O)(CCNC(c2cc(O)n(C)n2)=O)C1 N1(CC2CCN(C)C2)CCC(C2CCCN2C(c2ccnnc2O)C2CC2)CC1 C#Cc1cc(C(=O)NC2COCC2NC(=O)CCc2cnc(C)s2)ccc1Cl N1(C(C)CC2CC2)CCOCC(C(=O)NCCCOc2ccccc2Cl)C1 C1(F)(CNC(CSCCN(CC)CC)=O)COCCN(C(c2ncc(Cl)s2)=O)C1 CC1(C)OC2CN(S(=O)(=O)c3cccc(CC(=O)O)c3)CC2O1 c1(OC)ccnc(NC(C2CCCC2NC(c2cccc(F)n2)=O)=O)c1I CCC(CNC(C1CN(C)CCO1)=O)(CC)C(=O)N(C)Cc1ccccc1C C(=O)(C#CC1CCC(=O)CC1)NCC(C(C)C)NC(c1ncsc1C(F)(F)F)=O c1(C(N2CC(C(C(=O)NC3(N(C)C)CCC3)OC)C2)=O)ccc(COC)c(F)c1 c1(C(=O)NC2CC(C)(COC)N(C(=O)C=CCO)C2)cc(C)c(C)nc1C C(=O)(C(C)NC(=O)CN(C1CN(C(=O)CCC2CCCC2)C1)C)NC(C)C S(=O)(=O)(c1cc(Cl)c(Cl)cc1Cl)N1CC2CCN(C(CC(CC)O)=O)C2C1 N1(C(Cc2c(C)cco2)=O)CCCC(CO)(NC(=O)CC2CC(C)C2)C1 C1(C(N2CCC(CCCC)CC2)=O)CCc2nc(C3CC3)ncc2C1 C(=O)(C(C)(C)CC#N)NCC1CC(NC(C(C2CCOCC2)OC)=O)C(O)C1 c1(C(=O)NCCCN(C(C(C(=O)OC)OC)=O)CCO)[nH]nc([N+](=O)[O-])c1Cl C1(NC(c2cc(SC)oc2C)=O)CCCN(C(=O)CC2(O)CCCOC2)CC1 c1(-n2cc(C(=O)NCC(=O)NCC3(C#N)CC3)nn2)ccc(NC(N)=O)cc1 CCC(CC(F)F)C(=O)N1CCCCC1CCNC(C1CC2CCC(C1)N2C)=O C(=O)(CC(C)C(=O)OC)N1C(CNC(c2cnc(CC)s2)=O)COCC1 C(=O)(C1CCCn2cnnc21)N1CCCN(C(=O)CC2CS(=O)(=O)C2)CC1CO C(CCCC(CO)NC(C1(CO)CCCO1)=O)NC(c1n(C)ncc1)=O c1(OC)cccc2c(C(C)NC(C3CN(C(=O)C(F)(F)F)C3)=O)c(C)[nH]c12 n1(CC)nc(C(=O)NCC2CC2NC(=O)CC(O)C(C)C)c(=O)c2ccccc12 C=C(C)CC(C(=O)NCc1cccc(NC(c2cc(C)sc2N)=O)c1)OC c1(C(N2C(C)CC(NC(CCCCCC#C)=O)C2)=O)cc2cc(C)ccc2[nH]1 c1(SC)ccc(C(N2CC(NC(=O)CC3(CO)CC3)C3(CC3)C2)=O)c(Cl)c1 c1(C(N2CCC(CN(C(C(C)O)=O)Cc3cccnc3)C2)=O)ccc(F)cn1 CCC(CCC(=O)NC1(C)CCC(C)C1)NC(=O)CC(C)(C)COC c1(C(C(=O)N(C(c2ccccc2)C(=O)OCC)CCOC)F)cccc(Br)c1F N1(CCCN(C(=O)Nc2ccccc2)C2CC2)CCOCC1 CC1CCCC(CCNCC(c2ccc(O)cc2)O)C1 N1(C(CC=CC(C)(C)C)=O)CCC(NC(c2cccc(OC(F)F)n2)=O)CC1 c1(C(=O)NC2CCC(CCNC(C(N)=O)=O)C2)cccc(CCO)c1 N1(C(c2c(NC)scn2)=O)CCC(NC(C2CCC(C)(C)CC2)=O)C12CC2 c1(CN2CC(C)(CC(N3CC(C)N(C)CC3)=O)C2)cccc2c1OCC2 C1(NC(C2C(=C)CC2)=O)CCC2CN(c3cc(C(=O)OC)nc(C)n3)CC2C1 Cc1nc(C2CC2)oc1C(=O)NC1CN(C(C2(Cl)CC23CCC3)=O)CC1O.C1(C)CC1 CN=c1[nH]c(=NCC2COC(=O)N2)[nH]c(=NCCc2cncc(Br)c2)[nH]1 n1(CCN(C(C23CSC(C2)C3)=O)C2CC2)cc(C2CC23CC3)nn1 C1(CCCO)CCNC(=O)CCC(=O)N1.C1(C(=O)OC(C)=O)CCC(C)CC1 CC#CCC(C(=O)NOC(C)C(=O)OC)NC(=O)C(CC)CCCCC C(=O)(CC(C)(F)F)NCC(CCOC)NC(=O)C(c1cscc1Br)=O c1(CC)nc(C)ncc1C(=O)NCC1C(C)CCCN1C(C1CCCCN1C)=O C1(C(N2C(CNC(c3nc(-c4cn(C)nc4)sc3)=O)CCC2)=O)CCCC1(C)C C(CCC(O)C(=O)N(CC(N)=O)C)NC(c1c(CC)cns1)=O C=CC(C)(CC)C(=O)N(CCNC(c1cc(N)ccc1O)=O)Cc1ccccc1 N#Cc1cc(C2(C(=O)NC3COCCN(C(=O)OC(C)(C)C)C3)CC2)cc(Br)c1 Cc1cc(F)ccc1C(O)C(N1CCC(O)C(NC(=O)CSC2CC2)C1)=O N1(C(C(C(C)C)NC(N)=O)=O)CCC(NC(=O)C=Cc2ccsc2)C2(CCC2)C1 C1(CC(=O)NC(c2ccncn2)C)CCN(C(C2CC(F)C2)=O)C1 c1(OC)cc(NC(C2OCCC2CNC(C2CC(=O)NC(=O)C2)=O)=O)ccc1F N1(C(c2cc(C#N)sc2)=O)C2CCC1CC(NC(C1CC=CCO1)=O)C2 c1(C(C)C(N2CC(O)(CCNC(=O)C(C)c3ccon3)C2)=O)cc(F)cc(F)c1 C1(C(N2CCC(C)(CCNC(c3ccc(C(N)=O)o3)=O)C2)=O)(SC)CCOCC1 CC(C)C(N=[N+]=[N-])C(=O)N1CCC(N(C)C)C1.N12CCC(C1C)C(=O)NO2 N1(C(C2C(OCC)C2)=O)CCOCC(CNC(C2CCS(=O)CC2)=O)C1 c1(CC)n[nH]c(CC)c1CC(=O)NC1CC1CNC(=O)C=Cc1ccc(Cl)s1 c1(C(=O)NC2CC(CNC(CCSCCC)=O)C23CCC3)ccn2ccnc2c1 CCC(F)(F)C(=O)N(CC(O)CNC(c1cscc1C(F)F)=O)C C1(NC(c2cc(N)cc(O)c2)=O)CC(NC(=O)Cc2cnsc2)C12CCOCC2 c1(OC)ccc(F)cc1NC(C1CC1C(=O)NC1(CC#N)CCC1)=O N1(C(C2(F)C(C)C2)=O)CCC(N(C(=O)CNC(c2ccccn2)=O)C)C1 C1(C(=O)OC)CC(C)(NC(=O)CC2(NC(C34COCC3C4)=O)CC2)C1 N1(C(CCSCC)=O)CCC(CN(C)C(C2(C(=O)NCC)CCC2)=O)C1 CC(N=c1[nH]nc(O)s1)C1CCN(C(c2cc(C3CC3)nn2C)=O)CC1 C(C)(CCCCN=c1[nH]cnc2cc(C(=O)OC)ccc12)NC(CN(CC)CC)=O N1(C(c2c(C)cn(C)c2)=O)CC(C)N(C(c2cc(-c3ccoc3)[nH]n2)=O)CC1C CC1(C)COC1C(=O)NC(CNC(=O)CC1C=CCC1)C1CCC1 c1(C(=O)NCC(C)(C2CCC2)NC(C(F)=CCC)=O)nsnc1O C(=O)(C(O)CN1CCCC1)N1CC(C(C)(O)Cc2cccs2)C1 C(=O)(C(C)CCCC)N1CCN(CC)CC1.C(C(=O)NC)N(CC#C)CC C1(C(=O)NC2C(CC=C)COC2)CC2CN(C(=O)CC(C)n3cccn3)CC2C1 Cc1nonc1CC(=O)NC(CN(C(=O)C(O)CN(C)C)C)Cc1ccccc1 C12(C(=O)NC3C(OC)CC3O)CC(CN(C(c3cn(C4CC4)nn3)=O)C1)C2 n1(CC(=O)NCCCOCC)ccc(=NCc2cccc3ccn(C)c23)nc1O C(=O)(C(C)(C)C(C)(F)F)N1CCC(N(CCC)C(C2OCCC2CC)=O)C1 c1(-c2c(C)ccc(C#N)c2)ccc2c(c1)C1(CCN(S(=O)(=O)C3CC3)C1)C(=O)N2 c1(C(=O)NC(CC2CN(C(C(CC)F)=O)C2)C)cncc(NS(C)(=O)=O)c1 CC1CC(NC(=O)C(=O)NC2CC2)CCN1C(=O)C(C)CSc1ccc(F)cc1 c1(C(N2CC3C(NC(c4c[nH]c(=NC)s4)=O)(C3)C2)=O)n[nH]c2c1CC(C)CC2 N1(C(=O)OC(C)(C)C)CCC2CCN(Cc3cc(C4CC4)ccc3F)C2C1 c1(CNCC2(NC(C3C(C)C3)=O)COC2)ccc([N+](=O)[O-])o1 N1(C(c2ccc(CC)c(F)c2)C(=O)NCC(F)F)Cc2ccccc2CCC1C Cc1cccc(C)c1NC(=O)C(N1CCOC(C)(C(F)F)C1)c1ncsc1C c1(C(=O)NC2C3CC2CN(C(C2C4CCCC24)=O)C3)ccc2cc(Cl)ccc2c1 C1(C(N(CCCCC)C)=O)(NCC2CCC2)CCNCC1 N1(C(C2CC3C=CC2C3)=O)CCC2(CC1)CCN(C(C1CC3(CCO1)CC3)=O)C2 C1(C2CN(C(c3ccc(Br)cc3)=O)C2)(NC(Cc2nc(C)oc2)=O)CC1 CCCC(CCC)CC(=O)N1CC(O)CC1CNC(=O)CC1(CC)CCOCC1 c1(N(C(C2C(C)C2)=O)C(N2CCCC2C)=O)cc(Br)ccc1O C1(C(C)C)CN(C(c2cn(CCCF)nn2)=O)CCN1C(=O)COC1CC1 C1(NC(CC(CC)(C)C)=O)CCC2(CCCN(C(c3cc(Br)no3)=O)C2)C1 C1(C(N2CCN(C(C(CC=CC)(C)C)=O)CC23CC3)=O)CCc2ccccc2C1 c1(NC(=O)NC(c2cccc(Cl)c2)CC)nc2cc(C#N)ccc2o1 Cc1cc(C(N2CC(CNC(C3COC(=O)N3C)=O)C(C)(C)C2)=O)cc(O)n1 C=C1CCN(C(=O)C=C(C)CCC)C(C(=O)NC2COC3(CCC3)C2)C1 Cc1c(Cl)c(C(=O)NCC(=C2CN(C(=O)CC3OCCC3(C)C)C2)F)nn1C C1(C(=O)NCc2c(C)nn[nH]2)CN(C(C2(O)CCC2)=O)CCN1C C(CC1CN(C(=O)OC(C)(C)C)C1)(C(=O)NC(C)C)NC(CCOCC(C)C)=O C1(C(=O)NCC2(CCNC(CN(CC)CC)=O)CC2)CCCSC1 c1(OC)ccc(C)cc1CNCC1COCCN1C(=O)Cc1ccc(Br)[nH]1 c1(C(N2CCC(NC(c3cnn4cccc4c3)=O)C2)=O)c(F)cc(Br)cc1Br C1(C(N2CC(COC)(NC(c3sccc3F)=O)C2)=O)CC(C2CC2)=NO1 N1(CC(c2ccc(C)cc2)=O)CCC(O)(C(=O)NC2(C)CCCC2)CC1 n1(CC)cc(Cl)cc1C(=O)NCC1CCN(C(c2n[nH]c(C)c2Br)=O)CC1 c1(C(=O)NC(C2CCCCC2)C(=O)NC(CCCCC)C)c[nH]c(C#N)c1C CCC(C(=O)NCC(C)CN(C)C(c1ccc(C(F)(F)F)o1)=O)C(C)(F)F c1(C(=O)NCC2N(C(CCOCC)=O)CCC(C)C2)cc2c(nc1O)CCSC2 c1(CCC)cc(C(=O)NC2(C)CCN(C(c3coc(N(C)C)n3)=O)C2)n(C)n1 CCCCC(O)CC(=O)NCC1(CCNC(=O)C(CC)c2cccnc2)CC1 c1(OC)cccc([N+](=O)[O-])c1CN1CCNCC1C(=O)Nc1ccnc(C#N)c1 C=CC1(C2(C(=O)NCC3CC3CNC(=O)CCCC(CC)CC)CCC2)CCC1 c1(C(N2CC(C(C)NC(c3n(CC)nnc3)=O)C2)=O)cccc(C(C)C)c1 Cn1ncc2c1CN(C(=O)C(CC1CC1)NC(C1C=CCCC1)=O)C2 C1(NC(c2cn(CC)nc2)=O)C(C)CCN(C(=O)CCC2CCCOC2)C1C N1(C(c2ccc(C=C)cc2)=O)CC(C(N2CCC23CC(O)C3)=O)CC12CCC2 c1(C(=O)NCC(CCNC(c2cnc(C3CC3)o2)=O)O)occ2c1CCOC2 C(=O)(C(C(C)(C)C)NS(C)(=O)=O)NCC1N(C(CC(C)(C)C)=O)CC(F)C1 C1(c2cn(CCCC(=O)N(C)CC3(C)CCC(CO)O3)nn2)CCC(C)(C)CC1 N1(C(c2cc(C3CC3)cs2)=O)CCOC(CCNC(=O)C(F)(F)CC2CC2)C1 C1(NC(c2c(C)sc(O)n2)=O)CCN(c2snc(Cl)c2C#N)CC1C Cc1ccc(C(N2CCC(C)(C(=O)NCc3ncc(Br)s3)C2)=O)c(F)c1 C1(CC#C)(C(N2CC(CC(C)NC(c3cc(C)c(C)s3)=O)C2)=O)CCCCO1 C12(C(N(C)CC3(C)CCCC3NC(C3COCCO3)=O)=O)CCCN1CCC2 C1(C2(O)CN(C(C34CC(F)(C3)C4)=O)C2)(CNC(C2CC(C)SCC2)=O)CC1 C1(NC(C)=O)CN(C(=O)CC2(C3CC3)CC2)CCC1C(F)(F)F C1(C)(CC)CCCC(NC(=O)CC(c2ccc(OC)cc2)N)C1 c1(C(N2C(C)CC(NC(c3cc(C(CC)C)no3)=O)C2)=O)ccc(C)c(CO)c1 c1(N2CCN(C(C#CC(C)C)=O)CC(O)C2)ccc([N+](=O)[O-])c(OC(F)F)c1 c1(C(=O)OCC)c(C(C)(C)C)csc1NCCC1(C)CC(C)=NO1 N1(CCCC2CCC(=O)C2)CCC2(CCS2)CC1 C(=O)(CC(CNC=O)CC(C)C)N(CCC1N(C(C(CC#C)C)=O)CCCC1)C c1(COC(c2ncc(OC)s2)=O)nc(Cl)ccc1Br N1(C(C23CC(CN(C(C45COCC4C5)=O)C2)C3)=O)CC(O)C(O)C12CCC2 Cc1noc2ncc(C(=O)NCC(CO)NC(=O)CC3(O)CCCOC3)cc12 C(=O)(C(F)CCC(C)(C)C)NC(N(CC(c1cccnc1)N1CCCC1)C)=O N1(C(CC(C)(C)SC)=O)CCC(C2CCOCC2)(CNC(=O)C(C)CC2CC2)C1 C1(NC(COCCCCC)=O)CC(O)CN(C(C2(CC3CC3)CCCCC2)=O)C1 C(=O)(C(=O)C(C)(C)C)N1CCC(N(C(=O)CC2CCNC(=O)C2)C)C1 CC(CC(N)=O)C(=O)NCCNC(=O)CNC(c1ccco1)=O Cc1ccc(C(=O)NCC(=O)N(C2CC2)Cc2cccnc2F)cc1[N+](=O)[O-] c1(OC)ccc(C(N2CCCC(C(=O)N(c3cncs3)C3CC3)C2)=O)cc1I C1(NC(C2CCCCC(C)(C)C2)=O)CN(C(=O)Cc2ccsc2)C2CCCCC12 C1(C)(NC(C2C(OC)C2)=O)CCN(C(c2nn(C3CCOCC3)cc2C)=O)C1 c1(C(N2C(C)CC(CNC(C3CC(F)(CO)C3)=O)C2)=O)ccc(O)c(N=[N+]=[N-])c1 N1(C(C(CC)SC)=O)CC2(CC(NC(C3CC3C(F)F)=O)CO2)C1 C1(C(=O)NC(CCSC)C)C(C)OCCN1C(=O)C(CN(C)C)N(C)C C1(C(=O)NCC(COCC)NC(=O)CN2CCS(=O)CC2)CCCC(OC)C1 c1(C(=O)NCC(CNC(c2nc(CC(C)C)sc2)=O)CO)ccnc(C2CC2)c1 C1(CNC(=O)CNC(=O)CCF)(NC)CCN(CC(=O)Nc2ccco2)CC1 c1(C(=O)Nc2c(C)nc(Cl)cc2)cc2c(-c3ccc4oncc4c3)cncc2s1 N1(C(C2OCC(C)C2)=O)CCCC2(NC(=O)C=Cc3cccc(F)c3)CCCC12 N#CC1CC(CNC(=O)CC2CCN2C(=O)C(C2CCOCC2)F)C1 C1(CCC(=O)NCCN(C(C(C)n2cncn2)=O)C2CCCC2)CCN(C)CC1 Cc1ccc(C(=O)NCC2CC(C)N(C(c3ccc(F)s3)=O)C2)nc1O Cc1ccc(C=CC(=O)N(C)CC2CCCN2C(c2cc(C(F)F)cs2)=O)s1 c1(N2CCC(COC)C2)cc(NC(=O)C=CCN(C)C)c(F)cc1[N+](=O)[O-] CC(CN(C)C)CCC(=O)NCC1(C(=O)N(C)CCF)CC1 Cc1oc([N+](=O)[O-])cc1C(N1CCCC(CNC(c2coc(C#N)c2)=O)C1)=O CC1(C)CN(C(=O)C(C)(F)c2ccon2)CC1NC(C1CCCS1(=O)=O)=O Cc1cc(C(=O)NCC2CCC(NC(C3CC=CC3)=O)C2)c2nc(C)n(C)c2n1 N1(C(=O)C2=NOC3(CCC3)C2)CC2C3CCC(C2C1)N(C(c1sccc1F)=O)C3 S(=O)(=O)(c1ccc2[nH]c(=NC(C)C(C)CO)sc2c1)NCc1ncc(C)nc1 C1(C2CCCN(C(C3(C)COC(=O)C3)=O)C2)(NC(C2(N(C)C)CCC2)=O)CC1 C(=O)C(C)CC(C)CC.C1(=O)CC2(CC2)CN1.O(NC(=O)C1CCC1)CCOC N1(CC)CCCC(CNC(=S)Nc2c(-c3ccccc3)ncn2C)C1 N1(C(C(CN(C(=O)CNC(=O)C2CC2)C)O)=O)CC(CO)CC12CCC2 c1(C(N(C2CCC(NC(=O)COCC(C)(C)C)CC2)C)=O)cnc(S)nc1 c1(CC(=O)NC2CC(CNC(CCN(C)CC)=O)C2(C)C)c(C)nn(C)c1Cl N1(C(C)=O)CCCCC1C(=O)NC(CNC(c1cc[nH]c(=N)n1)=O)C1CC1 Cc1oncc1C(=O)NC(C)C(N1CC(F)(CNC(c2n[nH]cc2Br)=O)C1)=O Cc1ccc2snc(C(=O)N(CC(O)CNC(=O)CC3CC3(C)C)C)c2c1 c1(C2(CNC(C3(C)CCC(NC(c4cnsn4)=O)C3)=O)CC2)cc(F)ccc1F c1(C(=O)NCC(C2(O)CN(C(c3ncccc3F)=O)C2)(C)C)cc(F)ccc1F C1(OC)CCC2(C(=O)NC3CC(NC(=O)Cn4c(C)csc4=O)CC3O)CC12 Clc1cc2c(N3CCC(n4cc(-c5ccccn5)nn4)C3)ccnc2cc1Cl C(=O)(CCC(O)C(C)(C)C)NC(C1CCN(c2nnc(O)s2)C1)C N1(C(CCc2nc(C)sc2)=O)CCC2(NC(=O)CSCCC#N)CC2C1 C1(CCC(=O)NC2CC(O)C2)(NC(CNC(N)=O)=O)CCCC1 c1(C(C)NC(c2cnn3ccncc23)=O)ccc2c(c1)CC(C)O2 c1(C(C(=O)NCC)N(C2CC2)Cc2ccccc2Br)cc(C(=O)OC)ccn1 c1(CC(N2CCCN(C(C(C)OC)=O)C(C)C2)=O)ccc([N+](=O)[O-])cc1F C1(NCC2NC(=O)C3(C2)CCC3)CCN(Cc2ccccc2)C2(CCC2)C1 N1(C(CC2C(NC(C3(C(C)C)CC3)=O)CCC2)=O)CC2CCCCC2C1C c1(N(C)C)ccc(CNC(=O)CC(C)(C)N(C(=O)CCCc2cnn[nH]2)C)cc1 N1(C(C2(CC)CCOC2)=O)CCC(OCCNC(=O)Cc2cn[nH]c2)CC1 CC(O)(C(=O)NCC1CCCN1c1ccncn1)C(F)(F)F c1(N(C)C)cc(NC(=O)CC2CC(NCc3ccc(C(F)(F)F)nc3)C2)ncn1 C12(NC(C3C(C=C)OCC3)=O)CCC(CN(C(=O)C=CC(CC)=CC)C1)C2 c1(CC)nc(C)[nH]c1C(=O)NCC1CCCCN1Cc1ccccc1Cl C1(NC(c2cnc(OCC)nc2)=O)CCN(C(C2CCCN2C)=O)C12CC2 C1(NC(C2C(C)(CC)C2)=O)C2CC1CN(C(=O)Cc1ccccc1F)C2 CC1CC(NC(C2(CCF)CCOCC2)=O)CN1C(C1(c2ccno2)CCC1)=O Cc1nc(C(=O)NCC2C=CC(NC(=O)C(C)CC(C)(F)F)C2)c2ccccn12 c1(NCC2CC(NC(c3n(CC#N)ncc3)=O)C2)ncnc2scc(Br)c12 C(CC(C(C)C)NC(c1ccnn1C)=O)NC(C(C)OCC#C)=O C1(NC(=O)COCC2CCCC2)COCC1NC(=O)COCC1CC1 C1(C(N2CCN(CCNC(C(CN(C)C)O)=O)C(=O)C2)=O)CC2OC(=O)OC2C1 c1(C(=O)NCC2CC(NC(C=Cc3cn(C)nn3)=O)C2)ccc(N)cc1O C1(CC)CCCN(CC(=O)NCC(C)(O)CNC(C2(C3(C)OCCO3)CC2)=O)C1 [N-]=[N+]=NCCCCC(=O)N1CC(CCNC(=O)CCCCN2CCCC2)C1 CCCC(F)(F)C(=O)NCC1OCCC1C(=O)Nc1csc(C)c1 C(=O)(C(CC)CC(F)(F)F)N(CCC)CCNC(c1c(C)coc1C1CC1)=O Cc1cc(C#N)cc(Cl)c1NC(C1CCCN(C(=O)CCCS(N)(=O)=O)C1)=O CC1CN(C(C2CC3CCC2O3)=O)CC1NC(=O)CC(O)c1ccccc1 c1(C(=O)NC2CC(CNC(Cc3n(C)ccc3)=O)C2)cc(F)c(CO)c(F)c1 C(CS(=O)(=O)c1cccc(C(F)(F)F)c1)N(C(c1ccc(SC)s1)=O)C1CC1 c1(C(N2CCC(N(C(=O)CCOCC)CCC)CC2)=O)ccn2cnnc2c1 N1(C(C(c2ccnn2C)C)=O)CC(C)C(C)(CNC(C23CCC(C2)C3(C)C)=O)C1 c1(C(=O)NC(C2(O)CCOCC2)C)ccc2c(n1)CCCN2 N1(C(C2(NC(C3CN4CCC3C4)=O)CC(O)C2)=O)CCC2(CC1)CC2 C(c1ccc(C)o1)=CC(N1CCC(C(N2CCC(CCC)C2)=O)C1)=O O(NC(=O)C(c1cccnc1)NC(c1ccc(CN(C)C)[nH]1)=O)C(C=C)C c1(NC(C=CC(CC)C)=O)cccc(NC(c2cc(N(C)C)ccn2)=O)c1 CCCC(O)CC(=O)N1CC(NC(c2cccc(NC(N)=O)c2)=O)C2(CC2)C1 C=C=CC(C)C(=O)NCC1CCN1C(c1cncc(N(C)C)c1)=O N1(CC=C)CCC(NC(=O)C(CCNC(=O)CC(C)(C)O)OC)CC1 Cc1noc(C)c1C(C)C(=O)NC(C)C(C)(C)CN(C)C Cc1n[nH]c(C)c1CC(=O)NCC(=C1CN(C(c2cnc(C(C)C)nc2)=O)C1)F N1(C(CCc2ccn(C)n2)=O)CC2(CCCN(C(=O)CC3CCCC(O)C3)C2)C1 N1(C(c2cccc(C(=O)OCC)c2)=O)CC(NC(C23CC(CO2)C3)=O)CC(O)C1 N1(C(c2ncc(C)nc2)=O)CC2(CC(CC(=O)N(CCO)C3CC3)C2)C1 c1(CNC(C2CCN(C(CCN(CCC)C)=O)C2)=O)cccc(OC)c1 N1(C(C2(C)C(C)OCC2)=O)CCC2(CC1)CC2C(=O)NCc1nn[nH]n1 Cc1cc(F)ccc1C(F)(F)C(=O)NCC(C)N(C)C(c1ccnn(C)c1=O)=O N1(C(CCCOCCC)=O)CCC(C)(C)C1CC(=O)N(C1CC(C)CC(C)C1)C CC1CN(CC(C)(C)O)CC(C)N1C.c12ccnc(c1)NS(=O)(=O)C2 Cc1ccc2[nH]nc(C(=O)NCC3CCN3C(=O)CC3CC(F)(F)C3)c2c1 C1(c2nc(C(C3CC3)OC)nn2-c2cnn(C)c2)Cc2ccccc2N1C C1(NC(C(CC)OC)=O)CCCCCN1C(=O)C(C)S(N)(=O)=O c1(CN(C(=O)CC2CCCCC2N)C)cccc(Cl)c1Cl C(=O)(C1=Cc2ccccc2C1)N1CCN(CCNC(CCCOC(C)C)=O)CC1 N1(C(C(C)O)=O)CCC2CCCC(C1)N2C(=O)CCc1cccc(Br)c1F C(CS(=O)(=O)CC(=O)N1CC2CCC2(CC(=O)NCc2cnsc2)C1)OC C1(C(N2CC(C(=O)NC(c3cc(C)on3)C)(CC)C2)=O)OC2CCC1C2 N1(CCCC)CCCCC1C(=O)N(C)CC1(CNC(=O)CC2CCC(=O)N2)CC1 C1(C(N2CCC(CCCO)C2)=O)CN(C(=O)CC=C(Cl)Cl)CC12CCC2 CC1=C(C(=O)N(C2CCCCC2N(CC(=O)OC(C)(C)C)C)C)CC1 N1(C(C(C)C#N)=O)CCC2C(NC(C3(Br)CC3)=O)CC12 C1(NC(c2cc(C)nc(O)c2)=O)CN(C(c2c(C)ccn2C)=O)CC(C)(C)C1 Cc1ccn(CC(=O)NC(C)(CNC(=O)Cc2nnc(O)s2)CC(C)C)c(=O)c1 Cc1c(C(N2CCN(C)CC2CNC(=O)CC2CCOC2)=O)cccc1Br C(=O)(C(C)CC(C)C)Nc1cccc(NC(C(CC)(C)F)=O)c1 N1(C(CC2CCC(C)(C)O2)=O)CC2(CCCC2)C1C(N1CC2CC2C1)=O C(=O)(C1Cc2ccc(F)cc21)NC1CC(C)(NC(C(C(CC)CC)F)=O)C1 C1(NC(C(n2c(C)ncc2)C)=O)CN(C(C2CC(C#N)C2)=O)CC12CC2 N1(C(C=Cc2n(CC)ncc2)=O)CCN(C(=O)C(F)OC(C)=O)CC(O)C1 C1(C(N2CC(F)(F)C2C2CC2)=O)CC2CCC1N2C(C1COCC1C(N)=O)=O Cc1cccc(CNC(=O)C(C2CC2(C)Br)N(CC(=O)N(C(C)C)C(C)C)C)c1 CC1CN(C)CCCN1C(c1cc(C2CCOCC2)[nH]n1)C(=O)NC1CCCC1 C1(C(N2CC3CC(C(N4CCC4CC4CC4)=O)CC3C2)=O)CCC(C2CC2)CC1 C(CC(=O)N1CCOC2CC12)(C(C)C)NC(c1c(C)snc1)=O CC(C)C(F)(CNC(C1CC2CC1CC2=O)=O)C(=O)NC(C)C(O)C(F)F C#CCC(CC(=O)OC)NC(C1C=CC(NC(C2CCCSC2)=O)C1)=O C1(O)(C(=O)NCC=CCNC(C2N(CCC)CCC2)=O)CCc2ccccc2C1 Cc1ccc(F)c(C(C)NC2CCC(N)C2)c1F C1(CC(=O)NC(C2N(C(Cc3c(C)occ3)=O)CCC2)(C)C)CCS(=O)(=O)C1 Cc1cc(C(=O)O)cc(C)c1NC(c1ccc(C(F)F)c(F)c1)N(C)C C1(NC(C(=O)OC)C)CSC(C(F)(F)F)C1 c1(C(=O)NCC(C2CCCCC2)NC(C(C)(C)C)=O)sc(F)cc1Br C(CCCCCNC(C1CC(CF)C1)=O)NC(=O)CC1CCOC1 N1(C(C(CC)(F)F)=O)Cc2occ(C(=O)NCC(C)(C)CO)c2C1 CS(=O)(=O)c1cnc(NCC2CCCC2NC(c2c[nH]cc2Br)=O)c(Cl)c1 N#Cc1ccc(CN2CCC3CC(C(N4CC(O)C(F)C4)=O)C3C2)c(F)c1 C=CCC(F)(F)C(=O)NC1CCC(NC(=O)COc2cncc(Br)c2)C1 C12(C(=O)NCC(CC=C)NC(=O)CC3CC(C)(C)CO3)CCC(C#N)(CC1)CC2 c1(SC)nc(O)c(C(=O)N(C(C)CNC(c2ccc(Cl)s2)=O)C)cc1C#N CCCC(C)C(CO)NC(C1(CCNC(=O)CC2CCSCC2)CC1)=O N1(C(c2scc(OC)c2)=O)CC(OC)CC1CNC(=O)C(N1CCNC1=O)C C1(OC)(CNC(c2ccnc(Cl)c2F)=O)CCN(C(=O)C(=O)NC2CC2)CC1 c1(C(=O)OC)ccc(S(=O)(=O)NC(C)CCC2CCCCC2)c(OC)c1 C(N=c1ccc2cc(S(=O)(=O)O)ccc2[nH]1)C1CC(N)C(O)C1 C#Cc1cc(C(=O)NCC(C)(CO)NC(=O)C(CC)C2CCOCC2)cc(F)c1 C1(CNC(CNC(CC)=O)=O)CN(C(c2n[nH]c(C3CC3)c2C)=O)CCC1(F)F C1(NC(C(CCC)(C)C)=O)CC2CN(C(c3ccc(C#N)cc3)=O)CC2C1 CN1CCCC2(CCN(C(c3cncn3C)C(=O)NCCC#N)C2)C1=O N1(C(COCc2cc(OC)ncc2)=O)CCN(C(=O)CCCC(F)F)CC(O)C1 N=c1[nH]nc2ccc(N3CCN(C(=O)CCc4cc(Cl)cs4)CC3)nn12 C1(CNC(CC(=O)NCC)=O)CN(Cc2nnc(-c3cccs3)o2)CCCO1 C(=O)(N=c1ccn(C(F)F)[nH]1)C1(NC(C(C2CC2)OCC)=O)CCC1 Nc1ccc(-c2cn(CC(=O)Nc3ccccc3C(F)(F)F)nn2)cc1 c1(C(C)C)cccc(C(N2CC(Nc3cc(O)nc(C)n3)C(C)(C)C2)=O)c1F C1(S(C)=O)(C(=O)OCC)CCN(C(c2cc(C3CC3)nc3ccnn23)=O)CC1 C12(C(N3CCC(NC(c4ccoc4C(F)F)=O)C3)=O)CCC(CF)(C1)OC2 N1(CC2CC=CC(SCC)C2)CCC(CO)C(C)C1 c1(C(=O)OC)cc(C(=O)NCC=CCNC(C2(C(C)C)CCC2)=O)ccc1C C#CCC(CC(=O)NCC1CN(C(=O)C2CC2)CC1CC)c1ccccc1 C(=O)(CC(O)C(C)(C)C)NCC1(NC(C2N(C)C(=O)CC2)=O)CCCCC1 c1(C(=O)NC2(C(N3C(CNC(C)=O)C=CC3)=O)CC2(C)C)ncn(C)c1C C(=O)(CC(C)CC(C)C)NCC1CCN(C(C=C(C)Cl)=O)C(C)C1 C(=O)(CCC(=O)C(C)(C)C)N1CCC(C)(C(N(C)Cc2cnccn2)=O)C1 C1(NC(=O)C(C2(O)CN(C(=O)C=CCN3CCC3)C2)F)CC12CCCC2 C1(SC)CN(C(c2cc3c(Cl)c(Cl)ccc3[nH]2)=O)C2(CCCCC2)C1 c1(C(=O)NCCCNC(C=CC(=O)OCC)=O)ccc(OC)c(C)c1C CCC(C)(C#N)C(=O)NC1CC(O)(CNC(c2cnccn2)=O)C1 C1(C)(NC(C2C(CNC(CCc3n(C)ncc3)=O)CC2)=O)CCC2(CC1)CC2 C1(CNC(=O)C(c2ccc(Cl)cc2)CO)CCCN(C(=O)CC2CC(=O)C2)C1 C1(CC)C(NC(=O)Cn2ccc(C)c2)CCCN1C(=O)CCCn1cccn1 c1(C(=O)NCC2CCCN(C(CC(C)F)=O)C2)cc(N)c(F)cn1 C1(C(=O)OC)C=CCC1.c1(CCNC(C)(C)C)cnc[nH]1 N1(C(C2CCC(C)(F)CC2)=O)CC2CCCN(C(=O)COCc3nc[nH]n3)C2C1 n1(C(C)C)c(CSCCS(C)(=O)=O)nnc1Br N1(C(=O)C2CC2)CC2OCCN(C(=O)Cc3cnns3)C2C1 C1(NC(=O)C(C2CCN(Cc3c(C(=O)O)cccn3)C2)F)CC(=O)N(O)C1 CN1CC(OCCNC(=O)OCC(c2ccccc2)C2CC2)C(O)C1 N1(C(c2ccc(C)nn2)=O)CCC(CO)C(NC(c2coc3c2CSC3)=O)C1 c1(CC(=O)NC2(c3ccc(OC)cc3)CCOC2)cc(OC)c(OC)c(OC)c1 N1(C(CCC=CC)=O)CC(C)CCC1CNC(=O)C(N1CCC(C)CC1)=O C(=O)(C1CCCc2cncn21)N1CC2C(CNC(CCC#N)=O)(CCC2)C1 CC1CCC(=CC(N2CC(O)(CCNC(C3(Oc4cnn(C)c4)CC3)=O)C2)=O)C1 CC(CCC(=O)NCCN(C)C(C1CCS(=O)(=O)N1C)=O)S(C)(=O)=O C1(C(=O)NCC(=C2CN(C(C3CCC(c4cc[nH]n4)O3)=O)C2)F)(CC)CCOC1 c1(OC)ncc(C=CC(=O)NC2CC3(C2)CN(C(=O)CC2CC2(Cl)Cl)C3)cn1 c1(C(=O)NCCC2N(C(C(COC)O)=O)CCC2)ccc(C(C)C)cc1 C=CCCC(F)(F)C(=O)N(CCCCNC(c1cc(OC)cc(C)n1)=O)C C(C(=O)N(C(C)CC(=O)Nc1ccc(Cl)cc1)C)(C(C)C)SCC c1(NC(N)=O)cccc(F)c1C(=O)NCC1CC(NC(c2cnco2)=O)CCO1 N1(C(C23CCC(C)(CC2)CO3)=O)CCC(C2CC2NC(=O)C2=CCCC2)CC1 C1(C(C)C)CCC(C(=O)NC(Cn2cncn2)CC)N1C(=O)CC1OCCO1 C1(CC(=O)Nc2c(COC)cccc2)CN(C(=O)C(F)C(F)(F)F)CCC1C C12(CNC(C3(CC=C)CCC3)=O)CC1CN(C(C1(C(C)(C)O)CCC1)=O)C2 C1(C(N2CCC(OCCNC(c3c(C)cccn3)=O)C2)=O)COC(C)(C)CO1 c1(C(N2CC(CNC(c3cc(C)cc(O)c3)=O)OCC2)=O)cnc2ccoc2c1 c1(C(=O)NC2CCC(CNC(C=C(C)C)=O)CC2)cccc2c1N(C)C(=O)CO2 N1(C(C2CCN(C(=O)OCC)C2)=O)CCCC(N(C(=O)C(C)=C2CC2)CC)C1 N1(C(c2ncc(NC)nc2)=O)CCCN(C(c2ncccn2)=O)C(C(C)C)C1 C(CC(C)C)(C(=O)NCC1CCSC1)NC(Cc1cc(C)n(C)n1)=O C1(C(=O)NCC2(NC(C(C)S(N)(=O)=O)=O)CCCCC2)CCc2nc(O)[nH]c2C1 C1(NC(C(Cc2ccccc2)OC)=O)CCCCN(c2ncnc(=N)[nH]2)C1 N1(C(c2cc(CCC)c(C)s2)=O)CCN(C(C2CC2F)=O)C(CO)C1 N1(c2n(CCC=C)c(C34CCC(CC3)CC4)nn2)CCOc2c(C)cccc2C1 N1(C(C)C(N)=O)CCC(NC(=O)C(C)CCc2cccc(F)c2)CC(C)(C)C1 C1(C(=O)NC(C=CC(=O)N(CC(CC)(O)CC)C)C)CCCCC1(C)C c1(OC)ccc(N)c(C(=O)NC(C)CC(C)NC(c2ccncc2OC)=O)c1 c1(C(N2CC(CCCNC(COCC=C)=O)OCC2)=O)ccc(O)c(F)c1 c1(C(=O)NC2C(NC(C3CCC(C)(C)CO3)=O)C2)cccc2c1CNC2=O C(CCCC(C)NC(C1CC(CN(C)C)C1)=O)NC(C=CC(=O)OCC)=O C1(NC(c2c(C)n(C)nn2)=O)CC(NC(=O)C=C2CCOCC2)C12CCOCC2 C12(CC(=O)N(CC(O)CO)CCO)CC3CC(CC(C3)C1)C2.N12CC(F)(F)CC1C2=O c1(CCC(=O)N(CC(C)NC(=O)C=CSc2ccccc2)CC)ccccc1Cl Cn1ncc(=NC(=O)CC2CN(Cc3cc(Cl)ccc3O)C2)[nH]1 Cc1cc(C)cc(C=CC(N2CCOCC2CCC#N)=O)c1 Cc1c(C(N2CC(CC(C)NC(=O)C(C)CO)C2)=O)c(O)nc2ccccc12 c1(CN(C(CCOCCOC)=O)CCNC(c2cnc(C)s2)=O)ccccc1 C1(c2nnnn2C2(C)CC2)(NCCSC(C)C)CCC2CC12 N1(C(C(C)=CC)=O)CC(C)(C)C(NC(c2ccc(C(N)=O)o2)=O)C(C)(C)C1 C1(O)(C(=O)NCC(CC)(C)OC)CCCCC1O C1(CCNC(C2CC=CCC2)=O)CCCCN1C(=O)Cc1ccsc1Cl C1(C(N(C2CN(C(C(CCC)=CCC)=O)C2)C)=O)CN2CCC1CC2 C1(CC)CCCCN(C(c2cnc(CC(=O)Nc3ncc(C(C)C)o3)[nH]2)C)C1 C(C#Cc1cnn(C)c1)NC(CC(C(C)C)NC(C(COC)(C)C)=O)=O C1(CNC(C2=C(C)CCC2)=O)CCN(C(c2ccc3occc3c2)=O)CC1(F)F c1(OC)cc(C(=O)NCC(O)C(C)(C)O)ccc1OCCC(C)C C(c1cccc(O)c1)=CC(=O)NCC1CN(C(c2n(CC)ccn2)=O)C(C)C1 C(=O)(CCCCC(=O)N1CC(O)(CNC(C2CC(F)(CO)C2)=O)C1)NC N1(C(c2n(CC)cc(Cl)c2)=O)CC(NC(C2CC3C=CC2O3)=O)CC2(CC2)C1 N1(C(C(CN)SC2CCC2)=O)CCc2ccc(C(=O)O)cc2C1 C=CCC(C)(C)CC(=O)NC1CCC(N(C(=O)CCCCN(C)C(C)C)C)C1 C1(C(N(C)Cc2cc(OC)cc(F)c2)=O)CCn2cnnc2C1 N1(C(c2ccc(Cl)c(C)c2Cl)=O)CCOC2(CCN(S(=O)(=O)CCCl)CC2)C1 c1(CC(=O)NC(C)CCNC(C2CCCC2C)=O)ccc2c(c1)ncn2C Cc1cnc2c(C(N3CC(NC(c4nc(Cl)sc4Cl)=O)C4CC34)=O)cccn12 C1(C2(NC(CC(C)OC)=O)CC2)CCN(C(=O)CS(=O)(=O)N(C)C)CC1 C=Cc1ccc(C(=O)NC(CNC(=O)CCc2cccnc2)C(C)C)cc1 CC1CCN(C(c2cnn(CC(F)(F)F)n2)=O)CC1CNN(C)C1CC1 N1(C(C2(OCC)CCCCC2)=O)CCC2(CC1)CC2(C)C(=O)N(C)C(C)C C1(C)(C(N2CC(CNC(CCC3(C)CC3)=O)C(O)C2)=O)CCCS1(=O)=O c1(CC(=O)NCCN(C(C2N(C(CC)=O)CSC2)=O)C2CC2)cccc(Cl)c1 c12sc(nc1C)SC(CC)CN(C)C2=O.C(C)(C(=O)NCC(C)C)NC(C)=O C12(C(=O)NC(C3CCN(C(=O)CC4C=CCC4)CC3)C)C3C4C1C1C2C3C41C#N c1(CC(C)C)cc(C(=O)NC2CCC(CNC(c3csc(C(F)F)n3)=O)C2)n[nH]1 c1(N(C)C)nccc(C(=O)N(CC=CC(C)(C)C)CCO)c1Br C1(CN(C)C(c2cnc(S)[nH]2)=O)CCCC(NC(C2(c3ccsc3)CC2)=O)C1 CC(C)C(COCC1CCOC1)N=c1cnc(N(C)C)c[nH]1 C1(C(=O)NCCC(C)N(C(c2nc(OC)nc(O)c2)=O)C)CCC2(CCC2)CO1 c1(C(=O)NC(CC2CN(C(CCC(=C)Cl)=O)C2)C)oc2ccc(C)cc2c1C C1(NC(C(CC)C)=O)CCCCC12CCN(C(c1ccn(C3CCCC3)n1)=O)C2 CC1(CO)C=CCN1C(C1OCCC1CNC(C1CCCO1)=O)=O C1(NC(=O)COC2CCCCC2)CCCCCN(C(C2(C3CCCO3)CCC2)=O)C1 N1(C(C(CCC)(C)CC)=O)CCC2(C1)CN(C(C1(C)CCCCO1)=O)CCO2 N1(C(c2c(OC)scc2)C(=O)NC2CC2)CCCC(n2nc(C)cc2C)C1 N1(C(C(C)OCCC#C)=O)CCN(C)C(CNC(C2(n3cccn3)CCC2)=O)C1 c1(N2CCC(OCCNC(C=C(C)Cl)=O)C2)cc(Cl)ncn1 c1(C(N2CC(CN(C)Cc3ccsc3Br)C2)=O)c(I)ccnc1F C1(CC(N2CC(N(C(C(C=C)c3ccccc3)=O)C)C2)=O)CCCCCC1 C(=O)(CC(C)(O)C(F)(F)F)NC1CC2CN(C(CCC(C)(C)C)=O)CC1C2 Cn1ncc2c1CN(C(C1CC(F)(F)CN1Cc1cccc3nonc13)=O)CC2 CCCC(CNC(c1ccc(SC)o1)=O)C(=O)NC(c1nnc(O)n1C)C C1(NC(c2c(CC)occ2)=O)CN(C(C2(C)COC(=O)OC2)=O)CC2(CCC2)C1 CC1=C(C(=O)N2CCC2CNC(c2ccoc2CC(N)=O)=O)CCC1 N1(C(CCC2C(C)=NOC2=O)=O)CCCC(C)C1CNC(c1ccccn1)=O C1(C(N2CC(O)(CCNC(c3cncc(O)c3)=O)C2)=O)COCCC1(F)F Cc1cccc(NC(C2CN(Cc3ccc(I)cc3Br)CC(F)(F)C2)=O)c1C#N c1(C(=O)NCCC(C)N(C(C2CCC(CC)O2)=O)C)cc(C(F)F)ccc1Cl C1(N(C(C2CC=C(C)CC2)=O)C)CC2CCC(C1)N2C(=O)Cn1cnc(C#N)n1 N1(C(c2ccc(-n3cc(C4CCCC(O)C4)nn3)o2)=O)CCCC(O)(CO)CC1 C1(N(C(C(C)CC2CCC2)=O)C)CC2CCC(C1)N2C(=O)C(C)C(C)O n1(C(C)C)cc(C(=O)NC2CC2NC(=O)COC2CC=CC2)cn1 C1(COC)(CNC(=O)C=C(C)C)CCCN1C(=O)CCN1CCCC1=O N1(C(C2(C)COCCO2)=O)CCC2C(C(=O)NCC(F)C3CCC3)C2C1 CCCC(C)(CC)C(=O)NCCCNC(c1ccc(C#N)c(C)c1)=O N1(C(=O)C2=CCCOC2)CC2CCC1CN2C(c1cncc(Br)c1)=O c1(CCN(C(C)(C)C)C)cn(C(c2nccs2)C2CCN2C(C)=O)nn1 C1(CNC(c2[nH]cc(C)c2)=O)CCCCN1c1ccnc(C2CC2)n1 N1(C(C(C)CO)=O)CCC(C2CCN(C(=O)C3=CNC4=NCCC4=C3)C2)CC1 C1(N2C34CC(C3)(C4)C2=O)CCC2(CCNCC2)CC1.CC(C)(C)OC(=O)ON Cc1nc2cc(C(N3CCCN(C(C4(C(C)C)COC4)=O)CC3)=O)ccc2o1 C1(CC(=O)NCCCN(C(=O)CCNC2CCCC2)C(C)C)CCNC1=O C1(C(N2OCC(n3cc(C4C(SC(c5ccccc5)=O)C4)nn3)C2)=O)CCCC2(CCC2)O1 S(=O)(=O)(c1cnc(NCC2(S(C)=O)CC2)c(Cl)c1)N(C)Cc1cccc(F)c1F C(=O)(CC(C)(C)C(F)(F)F)N(CC(C)NC(Cn1c(C(C)C)nnn1)=O)C C=CCCC(C(=O)NCc1cc(O)cc(F)c1)NC(=O)CCc1ccco1 c1(OC)ncc(C(=O)NC2C=CC(CNC(=O)C3CC3)C2)cn1 N1(C(c2c(C)cc(CC)o2)=O)CC=C(C(=O)N2CC(COC(C)=O)C2)CC1 C1(NC(C2(C=C)CC2)=O)CC12CCN(C(=O)C(C)(C)N1CCCCC1)CC2 C1(OC(c2ccc(Cl)o2)=O)C2CC3C(=O)OC1C3O2 N1(C(c2ccc(C)cc2Cl)=O)CCN(C(=O)C(O)C(C)C)C(C)CC1C c1(C(N2CC3C(NC(c4c(COC)scc4)=O)(C3)C2)=O)ccc2sccc2c1 c1(C(=O)NC(CNC(C(C)NC(CC)=O)=O)(C)CC(C)C)ccnc2[nH]ncc12 C(C(C(C)C(C)C)NC(c1c(Br)c(C)nn1C)=O)NC(CCC)=O C(=O)(C1Cc2ccccc21)NC1(COC)CN(C(=O)CCc2ccsc2)C1 c1(C(=O)NCC(C)CNC(c2ccc3cncn3c2)=O)cccc2c1COCC2 C1(CC)CN(C(c2c(C)coc2CC)=O)CCN1C(C12CC(CC(F)F)(C1)C2)=O c1(C(=O)OC)ccc(NC2(F)CN(C(=O)COc3ccccc3)C2)c(I)n1 N1(C(CC(=O)NCC)=O)CCCC1(C)CNC(c1cn(C2CCOC2)nc1C)=O C1(CNC(C(n2cc(-c3ccnn3C3CC3(F)F)nn2)C)=O)CCC2(CC2)C1 c1(NC(=O)CCc2ncc[nH]2)cccc(NC(=O)C(O)CC2CCOCC2)c1 Cc1cc(=NCCOCC2CC2)[nH]c(NCC2CCCCC2c2ccccc2)n1 c1(C(N2CCC(NC(=O)COC(F)(F)F)CC2)=O)cc2c(O)cccc2[nH]1 C(N=c1[nH]c(=NC2CCC(C)C2)[nH]c2c1COC2)c1c(C)sc(Br)n1 N1(C(C(CC=CC)C)=O)CC(C)C(C)(C(N2CCC(c3cnco3)C2)=O)C1 S(=O)(=O)(c1c[nH]c(C(=O)N(CC(C)NC(=O)C(C)(C)C(N)=O)C)c1)NCCOC C1(=O)C(C)(c2ccccc2)CN1.Cc1ccc(C2CC2C(=O)NC2CC2)s1 Cn1ncc2cc(C(N3CC(NC(c4cccs4)=O)CCC(O)C3)=O)sc12 C(=O)(C(C)n1cncn1)NCC1(C(C)NC(CC)=O)CC1 C1(NC(C(CO)OC)=O)CN(C(C2(C)CCOC2)=O)CC1CO CC(C)S(=O)(=O)C(C)C(=O)N1CCCC(NC(c2ccn3ccnc3c2)=O)C1C C=CCC(C)C(=O)NC(CNC(c1n[nH]cc1C(C)C)=O)CC c1(C(=O)NCc2c(C(=O)NCCC3C(C)CCO3)con2)occ2c1CCC2 c1(C(N(C(C)CN(C(=O)Cc2nc(=N)[nH][nH]2)C)C)=O)ncc(F)cn1 c1(C(N2CCCC(F)(C(N3CCCCC3CCO)=O)C2)=O)ncn2c1CCC2 N1(C(C(C=CC)O)=O)CCC(CNC(c2cn(C(C)(C)C)nc2C)=O)C12CC2 C1(NC(CN2CCN(CC)CC2)=O)CC2(CCN(C(=O)C(C)=CC)C2)C1 C=C(C)CC(C(=O)N1CC(O)CC1C(=O)NC1CCC(C)CC1)OC C1(C(N(CCN(C(=O)CCc2cscn2)C)C)=O)CC1(F)F C1(OC)CC(C)CN(C(=O)CC(CC2CC2)NC(=O)C(n2nccc2C)C)C1 c1(C(=O)NC2C(C(=O)NCC3(O)CCC3)C2)ccc(Br)c(C(F)(F)F)c1 C(=O)(CC(C)C(C)(C)NC(=O)CC(C1CC1)C1CC1)Nc1ccc(OC)nc1 c1(C(=O)OC)cc(CCC(=O)NCCCNC(C2CC2F)=O)c[nH]1 C1(C(=O)NC(C(=O)OC)CC2CCCCN2)CNCCS(=O)(=O)C1 c1(OC)cc(C)cc(C(=O)NCC2(O)CC(CNC(=O)C(F)(F)C(C)O)C2)c1C c1(CN=C(NCC(CC)OC)NC(C)COC)nc2cc(C)ccc2n1C Cc1c(F)cc(C(N2CC(NC(=O)CNC(=O)CC(C)C)C(C)C2)=O)c(F)c1N C=CCC(C(=O)NC1CC(C(=O)NCC(F)C(C)(C)O)C1(C)C)C(C)C C1(C(N2CCC(OCC(N)=O)C2)=O)CC(O)CN1C(c1cnc(N)cn1)=O C1(CC)NC(=O)N(c2noc(C3(c4ccc(C5CC5)cc4)CC3)n2)C1=O CC1CCCC1(C)C(=O)N(C1CCN(C(=O)CCC(F)F)CC1)CCO N1(C(=O)NCC(C)(C)Oc2ccc(C)cn2)CC2C(=O)NC(=O)C2C1 c1(C(=O)NC2CC(CNC(c3c(C)nc[nH]3)=O)CC2O)cc(C(F)(F)F)c(Cl)cn1 c1(CC(C)C)ccc(-c2nc(CC(C)C)nn2-c2cnnn2C)cc1 N1(C(C(CC)OCC)=O)CCCC(C)(C)C1CNC(c1ccc2c(c1)COC2)=O C(=O)(C1CCc2nnc(C)n21)N1CC(NC(CC=CC)=O)C(OC)C1 Cc1ccc(NC(N2CCC(N(C)C(c3cnoc3C3CCC3)=O)C2)=O)cc1C c1(C(=O)NC2C(NC(CCNC(N)=O)=O)C2)cnc(O)cc1C(F)(F)F C(CC1OCCc2ccccc21)CN1C(C)(C)CC(Cc2ccccc2)C1 O=C(CC(C1CC1)C1CC1)NCCNC1CCN(C2CCCCC2)C1 CCC(C)(C)C(O)C(=O)N1CC(CC(=O)Nc2cnc(C)c(C)c2C)CC1(C)C c1(CCn2cc(CC(O)C3CCC3)nn2)cn2ccccc2n1 Cc1nc(O)c(Br)cc1C(=O)NCC1CN(C(c2cnsn2)=O)CC1C N1(C(c2cn3ccccc3n2)=O)CCOC2(CCN(C(C3CC4CC4C3)=O)C2)C1 N1(C(=O)C=Cc2ccco2)CCC(N2CCN(C(=O)CN3CCC3)CC2)CC1 C1(O)(C(C)NC(c2cc(C)nnc2)=O)CCN(C(=O)C(C)(C)CF)CC1 CCC(CC)C(F)C(=O)NC1(CNC(C2CCN(C)CC2)=O)CC1 N1(C(Cc2cc(C)nn2C)=O)CC2CCC1C1CN(C(=O)C=CC3CC3)CC21 n1(CC(=O)NC(CCNC(C=C(C)Cl)=O)C)ncn2cccc2c1=O c1(OC)c(C(C)NCC(=O)N(C)CC2(OC)CCC2)cccc1Cl c1(NC(N(C2C3N(C)C(CCC3)C2)C)=O)cnc2cc(Br)ccc2c1 c1(-c2ccc(N3CCCC(CNC(C(C=C)O)=O)C3)cc2)ncc2c(n1)CCC2 Cc1c(C(=O)Nc2nc3ncc(Cl)cc3s2)c(C)n2ccncc12 c1(N2CCC(C(C)NC(=O)Cc3cccn3C)CC2)cc(Cl)nc(S(C)(=O)=O)n1 Cc1ccc(COC(C)C(=O)NCC=CCNC(C2CCOC2(C)C)=O)cc1 CC1(C)CC(NC(=O)CC2CC3(CC3)CO2)CN1C(c1ccon1)=O c12cccc(c1)C2.c1(CC(=O)OC)cn(CC(=O)N(CC(C)C)C(C)C)nn1 c1(C(=O)NC(CC)(CNC(=O)CC2(OC)CC2)CC)cc(C)c2c(c1)CCC2 Cc1c(Cl)c(C(=O)NCC(C2CCN(C(c3cnn(C)n3)=O)CC2)C)nn1C N1(C(C(CCC)OCC)=O)CC(CNC(C2(F)CC2)=O)C(C)(C)C1 Cc1cc(Cl)nc(N)c1C(=O)NCCCCC(C)NC(=O)CSC(C)C Cc1cc(C)cc(S(=O)(=O)N2CCC=C(C(=O)NCCCS(C)(=O)=O)C2)c1 C(=O)(C1CCCn2nccc21)NC1CC(C)(NC(C(CCC)NC(C)=O)=O)C1 C1(C(=O)NCC(CSC)(C)O)CC(C)CCN1C(=O)CC(=O)NC1CC1 N1(C(C(=O)OC)c2ccns2)C(C)CN(CC(C)(C)C(=O)OC)CC1C Cn1ccnc1C(F)(F)C(=O)NC1CCOC1CNC(=O)CN1CCOCC1 C1(NC(=O)C(N2CCOC(c3ccccc3)C2)=O)CCN(CC(F)(F)F)C1=O C#CCCCCC(=O)N1CCCC1CNC(=O)CNC(=O)Cc1ccc(N)cc1 N1(C(CC=CC=C)=O)CC2CC(NC(C3CC34CCSCC4)=O)C(C2)C1 C1(C(N(CC)CC2CCN(C(=O)COCC(=O)NC)CC2)=O)CC(=O)OC1(C)C Cc1nc(Br)c(CNC2(c3nnnn3Cc3ccccc3)CC(C)N(C)C2)n1C c1(C(C(=O)NC(CC)C)N(CCCCN(C)C2CC2)C)ccc(OC(F)F)cc1 N1(C(CCC)=O)CCN(C(c2cn(C)nc2-c2ccoc2)=O)CC1C C1(NC(CCCc2scc(C)n2)=O)CN(C(C2C(C)(C)C2(C)C)=O)CCC1C C1(C(=O)NCC(C)NC(c2ncc3ccccn23)=O)CCCCC12OCCO2 N12CCN(CC1)C(=O)CNCC2.c1(SC(C)C(=O)N(C)C)nnnn1C1CC1 CCCC(C(O)C(=O)NCCC1CC=CCC1)NC(=O)COCCF c1(-c2cn(CCN(C)C(c3cnnc(O)c3)=O)nn2)cccc2ncccc12 c1(C(=O)NCC2OCCCN(C(C(=O)NCCOC)=O)C2)ccc(C#N)cc1F c1(C(=O)NC2CCCN(C(CCN(CCC)C)=O)C2)cc(NC(C)=O)ccc1C C(=O)(CS(=O)CCC(F)(F)F)N1CCC(O)(CN(C(=O)Cc2ccccc2)C)C1 N1(C(C(CNC(C(C)N(C(C)=O)C)=O)O)=O)CCC2(CC1)CC2CO C(=O)(C1=NOC(CNC(C2C3(CC3)C23CC3)=O)C1)NC(C)C(=O)NC1CC1 CC(F)(F)C(=O)NNC(=O)c1cccc(O)c1.c1ccc2occc2c1 c1(-c2cn(C(CNC(C3CC(=C)C3)=O)C)nn2)cc(C)cc(F)c1 C(N=c1cc(C)[nH]c(=NCCc2c[nH]nc2C)[nH]1)C1(OC)CCCOC1 CN1CC2CCC(C1)N2C(=O)CC(C1CC1)NC(C1C2CCCC(=O)C12)=O c1(C(C)=O)ccc(NC(=O)C(C)SCc2nc[nH]n2)cc1 N1(C(c2cnc(C)s2)=O)CC(NC(c2cccc(C(N)=O)c2)=O)C(C#N)C1 CC1(C)OCCC1CC(=O)NC1CCC1CNC(C1C(C)(C)C1(F)F)=O CC1(C)COC(C)(CNC(=O)C(=O)Nc2c(Cl)ccc(Cl)c2Cl)CO1 Cc1coc(C(N2CCC(NC(c3ccc(-n4ccnc4C)nc3)=O)C2)=O)c1C c1(NC(c2n(CCC)ccn2)c2nnnn2CCCF)cc(CC)c(F)cc1C C1(C(=O)NCC2C(C)=NOC2=O)CC2CC(O)CC(C1)C2.C12CCN1C(=O)N2 c1(NC(c2n(CCCSC)nnn2)(C2CCCCC2)C)cnc(C)c(Br)c1 c1(CC)c(C(=O)NC2(CN(C)C(C3CCC(F)C3)=O)CC2)cnc2ncnn12 C1(C(=O)NCC(CC(C)C)NC(=O)C=Cc2cnc[nH]2)CCCS(=O)(=O)C1 C1(CCNC(c2ccnnc2O)=O)CCN(C(c2ccnn2CC(F)F)=O)CC1 c1(OC)ncc(C(N2CC(NC(c3cc(C)ncc3C)=O)C(C)C2)=O)cc1C C1(C(N(CCCOC)CCO)=O)CCCCN1C(=O)CCc1nc(C)no1 NC1CC(CNCC2(c3ccc(F)cc3F)CCCC2)CCC1CO C1(CNC(CCC(C)N(C)C)=O)CCC(F)(CNC(C2CCO2)=O)CC1 C1(CCNC(C23CCC(C2)C3)=O)(NC(C2CC23CC3)=O)CCCC1 CC1CCC(=CC(=O)NCCC2(C(=O)NCC(C)OC(F)F)CCCC2)CC1 C1(c2n(C)cnc2)C(C(=O)NCCc2ccccc2C(F)(F)F)CC(=O)N1C1CC1 C=C=CCC(=O)NC(C)CN(C)C(c1cn(Cc2ccccc2)cn1)=O N1(C(C(C)NC=O)=O)CCCCC(CNC(=O)CCOCC2CC2)C1 C1(CNC(c2cnc(CC)[nH]2)=O)CN(C(C23CCC(CO)(CC2)C3)=O)CCC1C C1(NC(C2N(C(C(COC)OC)=O)CC(C)C2)=O)CC2C(O)C(O)CC12 C1(NC(c2ccnnc2S)=O)CC2CCCC(C1)N2C(=O)C(F)C1CCC1 N1(C(CN(C(C)C)C)=O)CC=C(CNC(C2CCC3CC3CC2)=O)CC1 O=S(=O)(c1nc(C(F)(F)F)cs1)N1CCn2nccc2C1 C(=O)(C1=CCCC(C)(C)C1)NC1CC(c2n(C)ncc2)OCC1 CC1CN(C(c2cc(C(F)(F)F)ccc2O)=O)CCCN1C(C1CC1(F)F)=O c1(NC(c2csc(-c3cnccn3)n2)=O)nccc2c(F)cccc12 C12(CC(F)(F)C1)N(C(C)C)C2=O.N1(C(c2ccccc2)=O)CCC(NC)CC1 CC1(C(=O)NC2COCCC2NC(=O)C=C2CN3CCC2CC3)CCCS1(=O)=O N1(C(C(C)O)=O)CCCCC(NC(=O)CSc2ccccc2Cl)CC1 c1(SCC(=O)N(CCN(C(c2cnnn2CC)=O)CC)CC)ccc(OC)cc1 c1(C(N2CC(C)(NC(CCC3CCC(C)O3)=O)C2)=O)c(O)cccc1Cl c1(SC)cc(C(N2CC3CC2(CNC(=O)C2=CCSC2)C3)=O)ccc1[N+](=O)[O-] C1(NC(C2N(CC)CC2)=O)CCN(C(c2nscc2Br)=O)CC1 c1(C(N(C)CC2N(C(C(c3cn(CC)nc3)=O)=O)CCC2)=O)cccn(C)c1=O N1(C(c2c(CNC(CCc3n(C)cnc3)=O)occ2)=O)CCCC2CC12 N1(C(=O)C2=CCCOC2)CC(NC(C2(C3CC3)CCC2)=O)CC2(CC2)C1 C(N=c1ccnc(N(CCC(C)(C)C)C)[nH]1)c1sc(CC)c(C)c1 C1(C(=O)NC2(C(N3CCC(CO)C(O)C3)=O)CCN(C)C2)CCOC(C)(C)C1 n1(CC(=O)NC2CCN(C(C3(O)CCCC3)=O)CC2O)ccc(=O)c([N+](=O)[O-])c1 c1(C(=O)NC2CC3CN(C(CCSCCC)=O)C2C3)ccc2c(O)n[nH]c2c1 N1(C(C(C)OCCCCCC)=O)CC2CCC1C1CN(C(=O)CCOC)CC21 c1(C(N2CCN(C(CC)=O)CC2C(C)C)=O)nsc2ccccc12 Cn1nc2c(c1C(=O)NC1CC3CC1N(C(c1ccnnc1O)=O)C3)CSCC2 C1(C(N2C(C)CN(C(C3CC4(C3)CC(O)C4)=O)CC2)=O)C2Cc3ccccc3C12 c1(C(=O)NC2C=CC(CNC(c3cc(C)oc3)=O)C2)ccncc1C(F)F CC1=NOC(C(=O)NCC2(CNC(c3cc(C)oc3C)=O)CCCC2)C1C C1(C(NOC)=O)CN(C(=O)CC2CC=CCN2C)CC1C(C)C Cc1nc(CC(F)(F)F)sc1C(=O)NCC1(C)CCN(C(=O)C2=CCOC2)C1 c1(OC)cc(C(=O)NCC(F)CNC(c2csc(Cl)c2)=O)ccc1Cl CCCCCC(O)C(=O)NCc1cccc(C(=O)NCC2CC=CCC2)n1 C1(N(C(C2CCCCC2O)=O)Cc2cc(Cl)ccc2F)COC2(CCNCC2)C1 C1(NC(C2C(=C)C2)=O)CC(OC)CN(C(=O)CSc2cccnc2)C1 Cc1ccc(C)c(C(N2CC3(CO)CC2(C(=O)NCc2cccc(F)c2)C3)=O)n1 c1(OC(C)C)ccc(C(N2C(CNC(C3CCCN3C=O)=O)CC3CC23)=O)nc1 C1(NC(c2cc(C)n(C3CC3)n2)=O)CN(C(c2cocn2)=O)CCC1C C#CCCCCCC(=O)N(C(C)(C)CC(=O)NC1(C2CCCCC2)CC1)C Cc1cccn(CC(=O)NCC2CN(C)CCN2C(=O)Cn2cc(Cl)cn2)c1=O C1(N(C(C)=O)Cc2cn(CCCNC(=O)NC)nn2)CCC(=O)NC1 n1(CC)nc(C(=O)NCCN(C)C(C2CCCN2CC(C)C)=O)cc1O C(CCC(=O)NCCc1nc[nH]n1)NC(C1C(C(=O)OC)C1)=O C1(CC)CN(C(=O)C(C)(C)CF)CCC1NC(c1ccn(CC#N)n1)=O c1(CNc2cncc(C(C)(C)O)c2)ccccc1S(=O)(=O)c1ccccc1 N1(C(c2c(CC)n(C)cc2)=O)CCCC(C)(C(N2CCCCC2)=O)C1 N1(C(CSC(C)C)=O)CC2CN(C(=O)C(C)C(C)(C)C)CC2(C)C1 C1(n2cc(C(C)NC(=O)CC3CCC(=O)O3)nn2)C2CC3C(C2)C13 c1(C(=O)NC(C(C)NC(c2ncc(C)cn2)=O)CO)cnn2c1NCC(C)C2 C(=O)(C(C)CC(F)(F)F)N1C(CNC(c2c(Cl)nc(OC)s2)=O)CC1 N1(C(CCc2onc(CC)n2)=O)CCN(C(=O)C(C)(C)N2CCCC2)CCC1C c1(NC(N2CCC(CC)CC2)=O)ccc2cnn(C)c2c1 C1(CNC(C=CCOC)=O)CC2CCC1N(C(=O)C1=CCCOC1)C2 CCC(O)C(F)(F)C(=O)N1CC2(COC(CNC(=O)CCCn3ccnc3)C2)C1 c1(CC(=O)NCC2CN(C(c3cnc(C(F)F)s3)=O)CC2O)ccc(F)cc1F C1(NC(C(CCSC)O)=O)CC2(CCN(C(C34CC(C(C)C)(CO3)C4)=O)C2)C1 C12(CNC(CC3C(C)(C)COC3)=O)CCCC1CN(C(=O)COC1CCOC1)C2 c1(C(N2CC3CC(NC(C4N=C(C)SC4)=O)C3C2)=O)cccc2c1NCCC2 c1(OCCCC)ccccc1C(=O)NCC12CC1CN(C(c1conc1C)=O)C2 CC(C)C(O)C(F)(F)C(=O)NC1CN(C(=O)Cc2ccon2)C2CCCCC12 c1(C(C)(C)C)cc(NC(=O)NCC2(C)CCOC2C2CC2)nc(Cl)n1 Cc1ncc(NC(=O)C(CC(F)F)N(C(=O)C(C)NC=O)C)cc1Cl C1(C(=O)NCc2scc(C)n2)(NC(=O)Cn2cc(Cl)cn2)CCC(C)(C)C1 c1(-c2c(CNCC(=O)NCCc3ccccc3)cccc2)cc(F)c(O)c(F)c1 C1(C(N(CCOCC=C)C)=O)N(C(=O)CCC(C)(C)C)CCC1(C)C N1(C(=O)Cc2ccc(F)cc2F)CC2CCN(C(C34CCC(CC3)O4)=O)CC2C1 CCC(C)(O)C(=O)NCC12CC1CN(C(c1coc(C(C)C)n1)=O)C2 Nc1ccc(C(=O)NC2CC(O)CN(C(=O)Cc3ccno3)C2)nc1N C1(NC(CSCCN(C)C)=O)CN(C(=O)CC2CN3CCN2CC3)CC(C)(C)C1 C#CC1(CNC(=O)C(C)(CO)NC(=O)C(CC)N(C)C)CCOCC1 C1(CNC(c2cc(F)n[nH]2)=O)CN(C(=O)CNC(C2CCCC2)=O)C2(CCC2)C1 Cc1cc(C(=O)NC2(CO)CN(Cc3ccc(Br)[nH]3)C2)cc(Cl)n1 CC1CN(C(C2(C)CCCOC2)=O)CCC1CNC(c1c[nH]ccc1=O)=O C12(CC)COC(C(N3CCCC3CNC(=O)C(c3ccc(Cl)cc3)(C)C)=O)(C1)C2 C(C(CNC(C1(CSC)CC1)=O)S(C)(=O)=O)NC(c1cnc(CC)nc1)=O N1(C(CCn2nc(C)c(Cl)c2C)=O)CCCC12CCCSC2 N1(C(=O)CCc2ccc(Br)c(F)c2)CCOc2ccc(Cl)cc2C1 C1(N(C(CC2(CNC(=O)CCn3ccnn3)CC2)=O)C)CCC(C(=O)OC)C1 N1(C(C2(CCOCC)CCC2)=O)CC2CC(NC(=O)C(=Cc3c[nH]cn3)F)C2C1 C(CC(CC)C(=O)NCCC1CCCN1C(=O)CSCC(F)(F)F)=CC N1(C(C(C(C)=O)(C)C)=O)CCC2(CC1)COC(C(=O)Nc1ncc(C)cn1)C2 C(N=c1[nH]c(=NCc2cccc(Cl)c2F)[nH]c2cc[nH]c12)c1c(F)cccc1F N1(C(c2cnnc(C)c2C)=O)CC2CCCC2(C(=O)NOCCC(F)(F)F)C1 c1(C(=O)NCC2CCN2C(=O)C=CC(F)(F)F)cnc2[nH]ncc2c1 c1(NCc2cc(C)ncn2)nc2ccccc2n1-c1ccccc1 C(c1ccc(F)cc1)=CC(N1CC(NC(CCCc2ncc(C)o2)=O)C(C)C1)=O CC#CCCCC(=O)N(CC(C)NC(C1CCCC(=O)O1)=O)C c1(-c2cc(C(=O)OC)ncc2)cc(C)c(S(=O)(=O)NCCCO)cc1C c1(C(=O)NC(CC=C)CNC(=O)CN2CC3CC3C2)cccc2[nH]ncc12 N1(Cc2c(C)cccc2)C(=O)CN(Cc2ccc(OC(F)F)nc2)C1=O C[Si](C)(C)CCCNC(=O)C(C1CCN(C(=O)CC(=O)NCC(F)F)C1)F N1(C(C(C)N(C)C(=O)C2CC2)=O)CCCC(F)(F)CC1 C(=O)(C(C)Cc1cccnc1)NCCC(C)NC(C1(C#N)CCC1)=O C(C)(C)(C(=O)NCC1(C(=O)NC2COC(Cn3cccn3)C2)CC1)N(C)C c1(C(N2C(Cn3cc(CN(C)S(N)(=O)=O)nn3)CCC2)=O)ccc(Br)cc1[N+](=O)[O-] N1(C(CC(C)CN(C)C)=O)CCCC(C)(CNC(c2cccnc2S)=O)C1 c1(C(C)NC(=O)NC2CC2C2CC2C)ccc(Cl)c(Cl)c1 c1(CC(=O)NCC(CC)(C)NC(c2cnn(CCF)c2)=O)cccnc1O C1(C(=O)NCc2c(OC)cccn2)C2CCC(C2)N1C(=O)CC1CCCC(=O)N1 CC1CN(C(=O)CONC(C2CCCN2C(C)(C)C)=O)CC(C)(C)CO1 CCC(F)(F)CC(=O)N1CCC(CC(N2CCCC2CC2CC2)=O)CC1 c1(CCC(=O)NC(C(C)NC(C2C(F)(F)C23CC3)=O)(C)C)ccccc1[N+](=O)[O-] C1(NC(C(C)OCC#C)=O)CCC(C)N(C(=O)COCCCC(C)C)C1 N1(C(c2cccc(OCC)n2)=O)CCCC(C(=O)NC2CC(N(C)C)C2)(SC)C1 N(C(=NCC1CCOC1)NCC(C)(C)OC(C)C)Cc1ccc(CC)s1 c1(C(=O)NCCC(CNC(C2C(=C)C2)=O)O)nc(O)nc(O)c1OC C1(c2nnnn2C)(NC(CCc2ccc(OC(C)C)cc2)C)CC12CCOCC2 c1(C(N(C2CCN(C(C3CCC(C)O3)=O)C2)CC)=O)c(C)nc2sccn12 n1(CCOC)nc(C(=O)N(C)CCN(C)C(c2ccc(Cl)cc2Cl)=O)ccc1=O c1(Nc2c(COC(c3nc(C(N)=O)sc3)=O)ccc(Cl)c2)ncc(Cl)nc1Cl N1(C(C(C)C)=O)CC2CCCC2(CNC(=O)C(C)Cc2cccnc2)C1 C(=O)(C1CCc2c[nH]nc21)NCC(C1CC1)NC(=O)CCCN1CCCCC1 Cc1cc(C(=O)NC(CNC(=O)CC2CC23CC3)C2CCC2)c2n[nH]cc2c1 C(CCCC(C)(F)F)NC(CN(C(=O)Cc1ccon1)CCOC)=O C1(NC(c2cc(C(N)=O)oc2)=O)CC(NC(=O)C(O)Cc2ccccn2)CC1O C1(C)(CNC(C(COC)OC)=O)CCCN1C(c1cc(C(F)(F)F)cs1)=O N1(C(COC)C(C)C)CCN(N2CCN(C3CCS(=O)(=O)C3)CC2)CC1 c1(C(C)(NC(=O)COC(F)F)Sc2ccc(F)cc2F)cc(C#N)ccn1 n1(CC)cnc2c1=NC1=NCC(=O)NC=2N1.C1(SCC2CC2)CN2CCC1CC2 C1(C2(O)CCC2)(CNC(C(C2CC(NC(c3c(C)n[nH]c3C)=O)C2)F)=O)CC1 c1(C(N2CCC(NC(=O)C=CCO)CC2C2CC2)=O)cc2ccccc2cc1F CN1N=C(CC(=O)N2CC(NC(c3ccc(O)nn3)=O)CC23CCCC3)CC1=O c1(C(C(=O)NC(c2ccccc2)C)N(CC(C)OC)C)ccc(Br)cn1 CC1(C(=O)NCC2CN(C(C3CCC(F)CC3)=O)CCCO2)CCCNS1(=O)=O C=CC1(C(=O)NC2CN(C(c3cc(CC)no3)=O)CC2C(F)(F)F)CCOCC1 C(C1CN(C(=O)C(COC)OC)CC1C(N1CCCC(OC)C1)=O)=CC c1(SC)ccc(Cl)c(C(=O)NC2CN(C(=O)Cn3nnc(=N)[nH]3)CC2C)c1 Cn1nc(Br)cc1C(N1CC(CNC(c2cn(CCF)nn2)=O)C(O)C1)=O CCCCCCCCCC(=O)NC1CCN(C(c2csc(C(C)=O)n2)=O)CC1O C=CC(CC)CC(=O)NC1(C2CC2)CCN(c2nc(C3CC3)nc(=N)[nH]2)C1 c1(CSC)cccc(C(=O)NCC(C)CNC(c2cc(Cl)c(Cl)s2)=O)c1 CCC(C)(CCC(C)C)C(=O)N1CC(F)(CNC(=O)CN2CC(C)(C)C2)C1 CC1CCC(O)CN1C(C1CCCOCC1)C(=O)NC1COC1 CC1CN(C(c2ncncc2F)=O)CC1NC(c1cn(CCCF)nn1)=O CC1(C)CCN(C(c2ccc(F)o2)=O)CC1CNC(=O)C(F)(F)c1ccccc1 C1(C)(CNC(CCC)=O)CC(F)(F)CN1C(=O)CCc1ccc(Cl)nc1 CC(C)(CCCNC(c1ncccc1C1CC1)=O)NC(=O)CSCC(N)=O c1(SC)cccc(C(=O)NC2CCCN(C(=O)CC(C)n3cccn3)CC2)c1Cl c1(C(=O)NC(C)CNC(C2CC3CC3C2)=O)cn(C(C)(C)C)nc1Br C1(CC)CN(C(C2CCCNC2=O)=O)CCN1C(=O)CCN(C)CC c1(C(=O)NC(C)CCNC(c2cc3n(c2)CCOC3)=O)cnn2c(N)ccnc12 N1(C(c2c(CC)cns2)=O)CCN(C(=O)CC2CCCC(C)O2)CC1 N1(C(C(C)O)=O)CCc2c(CNC(=O)Cn3cc(Br)ccc3=O)cccc2C1 Cc1ncc(C(=O)NC(C)CN(C(=O)CCc2csc(=N)[nH]2)C)c(C2CC2)n1 N1(C(Cc2c(C)n(C)nc2)=O)CC2CC(C1)C2NC(=O)C(c1cccc(F)c1)O C=C1CCC(C(N2CCC(C(=O)NC3CCN(C(C)C)C3=O)(C(C)C)C2)=O)CC1 c1(C(C(=O)NC(CNC(C2(COC)CC2)=O)C)C)c(C)noc1C C(=O)(CC(C)(O)COC)NC1C(NC(C2(CC)COC2)=O)CCC1 C(=O)(CCS(C)=O)N(C1CC(C(=O)NCC2(n3nccn3)CC2)C1)C c1(C(=O)NCCCC#C)ccc2c(c1)CN(C(c1ccoc1)=O)CC2 C1(CNC(C2C(C)C2(F)F)=O)CC(C)(C)CN1C(=O)C1=COCC1 N1(C(C2C(=C)C2C(=O)OC)=O)CCN(C(c2cc(C)ccc2O)=O)CC1C C1(CCC)CN(C(c2nnn(C(C)(C)C)n2)=O)CCN1C(c1cnc(C)nc1)=O N1(C(C(N(CC(=O)NCC2CC2)C)C2CC2)=O)CCC2(CNC(=O)O2)C1 C(C(F)(F)C(F)F)n1cc(C2N(C(C3(c4onc(C)n4)CC3)=O)CC2)nn1 C=C(Cl)CCC(=O)NC1CN(C(C2(COC)CCOCC2)=O)CC1C c1(C(=O)NCC(CNC(=O)CCOCC(F)F)OC)cnn(C)c1Cl c1(C(=O)NC2(CN(C(C3CC(C)OCC3)=O)C)CC2)cnn(C)c1C#N N1(C(CC=CCC)=O)CC2CCCC(NC(c3cnc4ccnn4c3C)=O)(C2)C1 c1(C(=O)NCC2(CCNC(C(C(C)O)N(C)C)=O)CC2)sc(C#N)cc1Cl c1(C(=O)NC2(C)CN(C(COCCCCC)=O)C2)cc(SC)ccc1Cl Cn1c2c(ccc1=O)C(NC(C1(C)C=CCCC1)=O)CCC2 O([Si](C)(C)C(C)(C)C)C(CC)CNc1ccc(Cl)cc1Cl C1(CNC(CS(=O)(=O)NCC)=O)CC2(CCC2)CN1C(c1c(Cl)cnn1C)=O N1(C(CCCNC(=O)OC)=O)CCC2CN(C(C3(C)CCC3)=O)CCC2C1 Cc1ccn2ncc(C(=O)NC3CC4CCC3N(C(C3(O)CCSC3)=O)C4)c2n1 N1(C(c2c(C)sc(Cl)n2)=O)CC2CCCC(NC(=O)C=CC3CCCCC3)C2C1 N1(C(CCC(=C)C)=O)CCC(C)C(CNC(c2ccc(N)c(C(C)=O)c2)=O)C1 C(=O)(CC(C)(C)C(F)(F)F)N1C(C)(CNC(c2ccc3c(c2)NCC3)=O)CCC1 c1(SCC(N2CCC(NC(c3ccn(C(C)C)n3)=O)CC2)=O)ccc(F)c(F)c1 N1(C(C(COCC=C)C(C)(C)C)=O)CCC(C2CC2NC(=O)CCC(N)=O)CC1 Cc1ccc(S(=O)(=O)NC2CCN(S(=O)(=O)c3cccc(Cl)c3F)C2)c(F)c1 N1(C(CCC(=C)Cl)=O)CCCC(C)(CNC(c2cccc(N3CCCC3)n2)=O)C1 C1(NC(C(C=C)O)=O)CN(C(C23CC4CC2C3C4(F)F)=O)C2(CCCCCC2)C1 N1(C(CN(C)Cc2ccccc2)=O)CC(NC(c2csc(CO)n2)=O)CC(O)C1 c1(C(=O)NC2(CCCNC(Cc3c(C)ocn3)=O)CC2)ccc2sccc2c1 C1(NC(C=CCCC=C(C)C)=O)CN(C(C2(CO)CC2)=O)CCC1CO Cc1nc(C2CC2)[nH]c1C(=O)NC(C)CCCCNC(C1CCCC12CC2)=O C1(NC(CCN(CCC)C)=O)(CO)CCCN(C(C2(C#N)CC2(C)C)=O)C1 C1(NC(C(C=CCCC)O)=O)CC(N=c2[nH]nc(-c3ccccc3)s2)C1 c1(CCC(=O)NC2CCN(C(c3cc(C(C)=O)sc3)=O)C2C)ccc(Cl)cc1F Cc1cc(F)ccc1-n1cc(C(=O)NCC2CCN2C(=O)C2=COCCC2)nn1 C1(C2CCN(C(=O)Cc3ccccc3CC(N)=O)C2)(NC(CS(N)(=O)=O)=O)CC1 C1(C(=O)NC(CNC(CCNC(=O)NC)=O)C)CCCN1C1CCCCC1 CCCCC(C)C(=O)N1CCC(C)C(CNC(c2cnc(O)cc2C)=O)C1 Cn1nc(C(=O)NC(C)(C(=O)NC2CC(O)C(O)C2)C2CCC2)cc1O C(=O)(CCCC(=O)N(C1(COCC)CCN(C(=O)C(C)C2CC2)C1)CC)OCC Cc1onc(C(=O)NC2CN(Cc3ccnc(F)c3)CC2F)c1C c1(C(N2CCC3(CN(c4nc(OC)c(F)cn4)C3)C2)=O)ccc2cnn(C)c2c1 c1(C(=O)NCC(C(C)C)NC(C(C)(C)OC)=O)cccc(NS(C)(=O)=O)c1 C(CN=C(NCCN1CCN(c2ccccc2)CC1)N1CCC(C)(OC)C1)OC N1(C(C(C(C)C)O)=O)CCC2CC(NC(c3cnn4ccncc34)=O)CCC2C1 c1(C(=O)NC2CC(CNC(C3C(C#C)C3)=O)C2)cc(C)c(Br)cc1C C1(CNC(c2cc(CCC)n(C)n2)=O)CC2CN(C(=O)C=Cc3cscn3)CC12 C(=O)(CCN=[N+]=[N-])N(C1CCCC1)CC(=O)NCC(c1cccs1)C CCC(CC)CCC(=O)N1CCC2(NC(c3cccc(OC)c3C)=O)CC2C1 C1(C)(CNC(C(C(C)C)O)=O)CN(C(=O)CCc2cccc(O)n2)CCO1 C1(CCC(=O)OC)CCC(NC(=O)CN2CC=CC2)C1.C12CCN1C2=O N1(C(c2cc(CC)sn2)=O)CC(NC(=O)CC(C)(C)C)C2(CCCC2)C1 C1(c2nnnn2C2CC23CCC3)(NCCCCCC)CC2CCC(C1)S2 C1(C(N2CCCC(CC)(CC)C2)C(=O)NCC2CCOC2)Cc2ccccc2C1 c1(C(=O)NCC2CN(C(CNC(=O)OCC)=O)C(C)C2)c(N)ccc(F)c1C N1(C(CCCCC(C)=O)=O)CCC2C(CCCN2C(c2coc(CO)c2)=O)C1 c1(CS(N2CC(C(C)NC(CCOC(C)C)=O)OCC2)(=O)=O)ccc(F)cc1F C1(OC(C2CCC(C(=O)OC)C2)=O)CC2CCC1CC21OCCO1 C(=O)(CC1OCc2ncccc21)NC(CCCNC(C=C1CCC(C)CC1)=O)C C(=O)(C(F)(F)C(F)F)NC1CC(CNC(Cn2nc(C)c(Cl)c2)=O)C1 O=C1NCC2(CO1)CN(C(=O)CC1CCCN1C(C1CC3CCC3C1)=O)C2 N1(C(c2c(CC)onc2C)=O)CCC2C(CCCN2C2CC2)C1 C(=O)(C(CCCC(C)C)NC(=O)C=C(C)C(C)(C)C)N1CC(SC)C1 C1(CC(=O)N(CC(C)NC(=O)C(C)(C)N(C)C)C)CC1C1CC1 N1(C(CC(C)c2ccccc2)=O)CCN(C(=O)C(F)CC2CCCC2)CC1 C(=O)(C(CCC)C(=O)OC)N(CC(C)NC(c1cnc(CCC)s1)=O)C c1(C(=O)NCC(CC)NC(=O)C(C2CC2)OC)cnc(O)c(C(C)=NO)c1 N#Cc1cccc(NC(C2CCCCC2NC(c2ccccc2CO)=O)=O)c1Cl c1(NC2CCC(NC(c3c(C)ncs3)=O)C2)nc(C(C)(C)C)nc(=N)[nH]1 n1(C(C=C)C)nc(-c2ccnc(Cl)c2)nc1C1CCN(C)C1=O CC1CN(C(=O)Nc2ccc(CN3CCN(C)CC3)cc2)C(C)(C)C1 C1(CNC(c2cc(C)n(C(F)F)n2)=O)CN(C(=O)CC2CC=CC2)CCCO1 C1(NC(CCc2ccn(C)n2)=O)CCCCC1CNC(=O)CC1CCCCC1O C(=O)(C(Cc1nonc1C)NC(=O)OC(C)(C)C)NCC(C)C Cc1nc(C)n(CC(=O)NCC2CCN(C(c3ccc(CC(C)C)nc3)=O)C2)n1 C(CCCC(=O)NC1CC1NC(=O)CC1CC2(CC2)CO1)OCC CC(CN=CC(O)C(O)CO)N(C)Cc1cccc(Cl)c1 CC1=C(C(=O)N2CCN(C(c3cncc(Br)c3C)=O)CC2C)C(=O)OC1(C)C C1(NC(c2cnn(CCC)c2C)=O)(CNC(=O)C2=CCCC2)CC2CCC1CC2 c1(OC)ccc(C(N2CCCC2CN(C)C(c2ccsc2OC)=O)=O)cc1F N1(C(COC2CN(C(=O)OC(C)(C)C)C2)=O)CC2CC3CC(C2)CC1C3 C1(C(N2CC3(C(NC(C4=CC(C)(C)C4)=O)CCC3)C2)=O)CNC2=C1CCCC2 C1(NC(C(C)NC(=O)NC)=O)CC2CCC(C1)N2C(c1ccc(C#N)c(Cl)c1)=O N1(C(CC(=C)C)=O)CCCC2C(NC(C3CC4(CSC4)C3)=O)C(C)(C)C12 C1(NC(=O)C2=COCCO2)CC2(CCN(C(c3n[nH]cc3F)=O)C2)C1 c1(C(=O)NC(CC)CNC(=O)CC2CC2(C)C)coc(C2CC2)n1 C(=O)(CCC1CCc2ccccc21)NCC1(C)CCCN1C(=O)CNS(N)(=O)=O Cc1cc(F)c(NC(C2CCCN2C(c2ccccc2CO)=O)=O)cc1[N+](=O)[O-] c1(C(=O)NC(CCCC)C(=O)NC(CCO)C2CC2)ccc2cncn2c1 Cc1ncc(Cl)cc1NC(C1(NC(c2cncc(O)c2)=O)CCN(C)C1)=O CC1CN(C(C2(CO)CC2)=O)CC(CCNC(c2n[nH]cc2Cl)=O)O1 Cc1c(C(=O)NCC2(NC(=O)CSc3nncn3C)CCC2)cncc1Cl c1(C2(CNC(c3n(CC)cnn3)c3nnnn3C)CC2)ccc(F)c(F)c1F C(=O)(CCCC(F)(F)C(F)(F)F)N1CC2(N(C(CC(CC)SC)=O)CC2)C1 c1(C(=O)NCC(CN(C(C(CC(C)C)OC)=O)C)C)ccc(C)c(Br)c1C C(=O)(C(C(C)C)C1CCC1)NCC1(NC(C(C)NC(=O)OC)=O)CCOC1 c1(OC(c2cc(Br)c(OCCO)s2)=O)cnnc(I)c1 CCC(CC)CCC(=O)NC(CC)CC(=O)N(CCCN1CCCC1)C c1(C(=O)NCC(CC=C)NC(=O)C(C)OC)ncc(C2CC2)cc1F C(C(CNC(c1ccnn1CCCC)=O)C(F)(F)F)NC(C(C=C)O)=O c1(C(N2CC(N(C)C(c3cc(Cl)cn3C)=O)C(F)C2)=O)cc2n(c1)CCC2 c1(C(=O)NC(C2CCN(C(c3c(C)nc(CC)o3)=O)C2)C)cc([N+](=O)[O-])oc1C c1(C(C)(C)C)cccc(C(=O)NC2(C)CC(NC(C3CCC(O)C3)=O)C2)n1 C1(CC(=O)N(CCCC)C)C(C2CC2)CCN1C(=O)Cn1cccc1 C1(C(C)CCO)CCCCN1C(=O)Cn1cc(CCN(C(C)(C)C)C)nn1 N1(C(c2csc(C)c2C)=O)CC2(CCN(C(=O)C(C)(C)c3cnco3)C2)C1 C1(N(C(CC(C)N(C)C)=O)CC2CC2)CCN(C(=O)C2=CCSC2)CC1 c1(OCC(=O)NC(CC)CNC(=O)CNC(=O)OC)ccccc1C C=CCCCCC(=O)N(C1CCCN(C(c2csc(C(F)F)c2)=O)C1)CCO C(=O)(N=c1cc[nH]c(CCO)c1)C1SCCN(C(c2cc(C#N)cc(Cl)c2)=O)C1 c1(CN2C(C(N3C4CCC3CC4)=O)C=CC2)cccc(Br)c1Br c1(C(N2CCOCC2CCC#N)C(=O)NCCC#N)cccc2c1nnn2C c1(C(C(=O)NCSc2ccc(F)cc2)N(C)C)cc([N+](=O)[O-])ccc1C#N C(=O)(C(CCOCC)NC(=O)CC(CC)OC)NCc1[nH]nc(CC)n1 CC(C)CC(CC(=O)NCC1CCCC1(C)C)NC(=O)C=Cc1cc[nH]c1 Cc1sc(O)nc1C(=O)NC1CC(C(=O)NC(C)CCC(C)C)C1 C(CCC(C)C(=O)N1CC(CNC(c2ccc(C)c(C)n2)=O)C(F)(F)C1)OC C1(C(=O)NCC(CO)NC(C2CC(=C3CCC3)C2)=O)(OC)CCC1 c1(OC)ccc(F)c(C(=O)NC(CNC(c2cc(Cl)cc(Cl)c2)=O)CO)c1N C(CCC(O)C(=O)NCC1(CN=[N+]=[N-])CC1)NC(c1cnn(C)c1Cl)=O C1(O)(CN(C(CN(CCOC)C)=O)C)CCN(C(=O)CC2(OC(C)C)CCC2)C1 C12(C(=O)NCCN(CCCN(C)C)C(c3ccc(F)cc3F)=O)CC1COC2(C)C N1(C(c2c(OC)ccnc2)=O)CC(C)(C)CC1CNC(=O)C(C)C(C)O CC1CN(C(c2cccc(O)n2)=O)CCC1CNC(=O)CC(C)(C)C1CC1 C1(C(=O)NCC(C=C)(C)C)C(CC)CCN1C(=O)C(C1CC1)OCC C1(CS(=O)(=O)N(CC(C)NC(C2CCOC2)=O)C)(C(F)(F)F)CCCC(=O)N1 C(=O)(CC1=CCN(C)CC1)NC1CN(C(C=C(COC)C)=O)C(C)CC1 N1(C(C2N(C)CC2)=O)CCCC(CC(=O)NCCC2CC(F)C2)C1 c1(OC)cc(C(=O)NC2(C)CCCN(C(c3ccc(C)nc3)=O)C2)cc(Br)c1 NS(=O)(=O)CC(=O)NCC1CN(C(c2csc(-c3ccoc3)n2)=O)CCO1 n1(CC)cc(C(=O)NCCC2(NC(c3coc(Cl)c3)=O)CC2)c(C(C)(C)C)n1 c1(C(N2CC(C(N)=O)OC(C)C2)C(=O)NCC)c(F)cc(Br)cc1F c1(-c2n(C)ncc2)ccc(S(=O)(=O)N2CCSC2CO)cc1 C1(NC(CC2(C)CCS(=O)(=O)N2)=O)CC2CCC(C1)N2C(=O)C(F)C1CCOC1 c1(C(=O)NCCC2CCC(NC(C3CCC=CCC3)=O)C2)ccnn2ccnc12 C1(C(C)C)CN(C(c2cc[nH]c2)=O)CCN1C(c1ccc(-c2cnccn2)s1)=O c1(CC(=O)NC(C2(CNC(c3[nH]cc(CC)c3)=O)CC2)C)ccnc(F)c1F CCCC(F)(F)C(=O)N(CCCCCC(=O)Nc1cnc(SC)nc1)C N1(C(C(C=C=C)C)=O)CCC2(CC1)C(NC(c1csc(Cl)c1)=O)CS2(=O)=O CC(C)CCCCC(=O)N1CC2(CO)CC1(C(=O)NCC1(O)CC1)C2 c1(CC(C(=O)N(C2CCN(C(c3cnc(OC)s3)=O)C2)CC)O)ccc(F)cc1 c1(N2CC(O)(CCNC(c3c(C(C)(C)C)ocn3)=O)C2)ncnc2c1CCO2 C1(C(=O)NCC2CN(C)C(=O)C2)CN(C(=O)C#CC2CCC2)CC12CC2 c1(N2C(=O)CC(NC(C(C(C)C)C3CCC3)=O)C2)cccc(C#CCO)c1 C1(SC)CN(C(=O)CNc2nccs2)CC1n1cc(CCS(N)(=O)=O)nn1 c1(C(N(CCC(C)NC(C2CCCCS2)=O)C)=O)cccc2ccsc12 c1(C(N(CCCNC(c2cnc(O)o2)=O)CC)=O)csc([N+](=O)[O-])c1 C1(C)(NC(c2c(C(C)NC(=O)CCN(C)C)noc2)=O)CN2CCC1CC2 C=CCCCCC(=O)NCCC1C(C)CCCN1C(c1cc([N+](=O)[O-])n[nH]1)=O C1(C(N2CC(C(=O)NOC3CCCC3)(SC)C2)=O)CC(C2CC2)=NO1 C1(C(N(C2CCN(C(=O)CCOCC3CC3)C2)CCC)=O)CC(C)CCO1 C1(C)(NC(C)C(C(=O)OC(C)(C)C)N(C)C)CCC(C)(C)CC1 Cc1cc(N)c(C(N2CCC(CCNC(=O)C(O)CCC(C)C)C2)=O)c(F)c1 C=CC(C)(O)CC(=O)NCC(C)(CNC(c1sc(C2CC2)nc1C)=O)OC c1(C(C(N2CC(CCC)C2)=O)OC)c(F)cc(Br)c(F)c1F.C(C)(C)(C)OC=O C(=O)(C(C)N(OC)C(=O)c1ccc(CNC(=O)CC2CCSC2)nc1)OC CC(C)(O)C(F)(F)C(=O)NC1COC2C(NC(c3n[nH]cc3[N+](=O)[O-])=O)COC12 N1(C(C2(Cl)C(C)(C)C2)=O)CC(OCc2ccccc2)C(F)(F)C1 C1(C(=O)NC(C2CCN(c3ncc(Br)cn3)CC2)C)CN(C)CC(C)O1 CN=c1[nH]cc(C(N2CC(NC(=O)C(c3ccccc3)C)C(O)C2)=O)o1 C1(CC(=O)NCC=CBr)CCCC(NC(=O)CC2CCOCC2)C1 C1(CNC(=O)CCc2ccc[nH]2)OCC2CCN(C(=O)C(F)Br)CC12 c1(-c2nc(CCCSCC(C)C)on2)ccc(C2CC2)cc1F.c1ccc(F)cc1 N1(CCN(C(C2CC(CC)C2)=O)C)CCN(C(=O)C(C)NC2CC2)CC1 C1(NC(C2CC2C(F)F)=O)CCC2(CC1)CN(C(C1CC13CCCC3)=O)CCO2 N1(CCCCOC)CCCC(C2CCCCN2C(C2CC2(C)C)=O)C1 CC(C)C(C(=O)NC1CC(NC(C2C(F)(F)C23CC3)=O)C1)c1cccnc1 C1(CNC(C2(C)C=CCCC2)=O)CCCCCN1C(c1ccc[nH]1)=O c1(CC)cc([N+](=O)[O-])ccc1NC1CN(C(C2CC23CCOCC3)=O)CC1C c1(OC)cnc(F)c(C(=O)NCCCC(C)NC(=O)C(C)(C(C)C)OC)c1 C1(C(=O)OCC)CN(C(c2ccnn2COC)C)CC1(C)C(F)F c1(C(=O)NC2CC3CN(C(C(C)(O)C4CCC4)=O)C2C3)ccn2ncnc2c1 c1(C(N(CC(CN(C(=O)C(F)C2CCOC2)C)O)C)=O)nc[nH]c1C(F)(F)F N1(C(c2c(CCC)n[nH]c2)=O)CCCC(C(N2CCC(F)(CF)C2)=O)C1C N1(C(CNC(CNC(C)=O)=O)=O)CC(NC(c2ccc(C)nn2)=O)C(F)C1 c1(C(C(=O)NCC(=C)C)N(CCC(C)C)C(C)(C)C)cc2ccnc(Cl)c2s1 C1(NC(C(c2ccnn2C)C)=O)CN(C(c2nc(Cl)ccc2N)=O)CC1C1CC1 C1(C(=O)NC(CCN(C(c2cn(CCC)nc2)=O)C)C)CC2CCC(C1)C2O C1(O)(CNC(CCOCC(C)C)=O)CCN(C(C2CCCC23CCC3)=O)CC1 C(CCC(F)(F)F)(C(=O)NC1CC1)NC(=O)CCOC1CC1 C123CCC(CC1)(CC2)CNC3=O.CC(C)(C)C(O)C(=O)NC1CCC(C)(O)CC1 c1(C(=O)NC(CCNC(C2(OC)CC2)=O)C)cc(Cl)cc(Cl)c1[N+](=O)[O-] N1(C(CCOCC#C)=O)CCN(C(c2ccc(N)cc2OC)=O)C(C)C1C C1(C(=O)NCCC2(C)CCN(C(=O)Cc3nncn3C)C2)(OCC)CCSCC1 C(CCCCC(=O)N1CCC(C(C)NC(=O)CCc2csc(=N)[nH]2)C1)OC C1(OC)CCNCC1C(=O)NCC(O)CCc1ccccc1 c1(CN2C(C)(C(=O)Nc3cccc(NC(=O)OC)c3)CC2)cc(F)c(F)c(F)c1 c1(OC)ncc(C(N2CCCc3c(CN)cccc32)=O)c2ccccc12 C(CC1CC1)(C(=O)NCC(O)CCNC(c1csc(CC(C)C)n1)=O)OC Cc1cc(Cl)cc(Br)c1NC(C1CC(F)(F)CN1Cc1cc(Br)cc(Cl)c1F)=O C1(NC(C2CCCN(CCC)C2)=O)CC2(CCN(C(c3cc(=O)n(C)o3)=O)C2)C1 C(C)(C)(CC(F)C(=O)NCCOC(=O)C1CC1)NC(C1C(C)CC(=O)CC1)=O N1(C(C(COC)N(C)C)=O)CCN(C(c2cc(OC)ncn2)=O)CC(O)C1 Cc1ccc(N)c(C(=O)NC2CC(CNC(C3(CO)CC3)=O)C2)c1F C1(N(CCC(C(=O)O)c2cn[nH]c2)C)CC(C(=O)O)N(C(=O)OC(C)(C)C)C1 N1(C(CSCCC)=O)C(CNC(c2cnn(C)c2COC)=O)CC2COCC12 N1(C(C(C)C)=O)CCN(C2CCN(C(c3csc(CC(F)F)n3)=O)CC2)CC1 c1(OC)ccc(Cl)cc1C(=O)NC1CC2(C1)CC2NC(c1[nH]c(C)nc1C)=O CCC(CC(=O)NC(C1CCN(C(=O)Cc2sc(S)nc2C)C1)(C)C)SC N1(C(c2n(C)nnc2)=O)CCC(C2CN(C(c3ccc(C4CC4)cn3)=O)C2)C1 c1(CC(C(=O)Nc2n(CC)nc(CN)c2)N)nccc2ccccc12 c1(C(N2CC(O)(C(C(=O)NCC3CS(=O)(=O)C3)F)C2)=O)c[nH]nc1[N+](=O)[O-] CC1=C(C(=O)NCC2CCN2C(c2cnc3n2CCCC3C)=O)S(=O)(=O)CCO1 c1(N(C)C)cccc(C(=O)NCC2N(C(C3CC4C=CC3C4)=O)CCC2)c1 Cc1ccc(C(=O)N(C2CC(C(=O)NCc3cnccc3Cl)C2)C)cc1F C1(CC(=O)N(C2CCN(C(c3cc(C)n(C(C)C)n3)=O)C2)CC)CC2CCC1C2 CCC(CCC(=O)O)NC(C1CCC(NC(=O)OC(C)(C)C)C1)=O CCCC(C(=O)N(CC(C)C(=O)NCCOC(C)=O)C)OC C1(C(=O)NC(c2ccncn2)(C)C)CCCN(C(=O)C=C2CCCCC2)C1 CC1CCC(C(=O)NCC23CC(CN2C(=O)CC2CCC24CCC4)C3)CC1 N1(C(Cc2c(C)noc2Cl)=O)CC2(CCCC2NC(=O)Cn2nnc(=N)[nH]2)C1 CN(C1C(=O)Nc2ccc(F)cc21)CCCOC1CCOC1 CC(CC(=O)NC1(C2CCCN2C(=O)CN2CCCC2=O)CC1)c1cnn(C)c1 C1(OC)CC(NC(=O)CCc2cnoc2)CN(C(c2coc(C(F)(F)F)c2)=O)C1 c1(C(=O)NCC2(NC(C(CC(C)C)O)=O)CCC2)cc2c(s1)CCC2=O C(CC(C)N=c1[nH]c(N2CCCCCCCC2)nc2ncn(C)c12)SC C=CCC(C(=O)NCCCCCNC(c1ccnc(OC)c1)=O)C(C)C Cc1cocc1C(=O)NCC12CC(NC(=O)C(C)NC(N)=O)(C1)C2 C12(NC(C3(CN(C)C)CC3)=O)CCC(CC1n1cc(-c3ccc(Cl)cc3)nn1)C2 c1(C(N2CCC(C(=O)Nc3nnco3)C(O)C2)=O)c(O)c(Cl)cc(Cl)c1Cl S(=O)(=O)(c1cccs1)NC(C1CCN(Cc2cc(OC)ncc2)CC1)=O C#CC1CCCCN1C(C1(C)CN(C(C2CC2Cl)=O)CC1C)=O C(C(C)(C)C(=O)NC(C)CCN(C(=O)CCCN(C)C(C)=O)C)OC N1(C(C2CN(C(C)=O)C2)=O)CCC2C(C1)NC(=O)CN2C(C1CCC12CCC2)=O CN=c1[nH]c(=NCc2nncs2)[nH]c(=NCc2ccc(F)cc2Cl)[nH]1 c1(C(=O)NC2CC3CN(C(c4c(C)n[nH]c4)=O)C2C3)c(F)ccc(F)c1F N1(C(c2nccc(C3CC3)n2)=O)CC(c2cn(Cc3c(C)ocn3)nn2)C(C)C1 C1(CC)CN(C(=NCCCCl)NCCSc2cc(Cl)ccc2Cl)CCS1 c1(C(N(N2CCCC(NC)C2)CC)=O)cc(OC)nc(OC)c1.n12cc(nn1)C2 CP(C)(=O)c1cnn(CC(=O)NCC(C)(C2CC2)NC(c2sccc2Cl)=O)c1 c1(C(=O)NCC2CN(C(CCc3cnc(C)o3)=O)C(C)C2)cccc2ccoc12 c1(CC(=O)NC(CC)COC)ccnc(O)c1 C(CC(C(C)(C)C)NC(c1cc2n(n1)CCC2)=O)N(C)C(C1CCC2(CC2)C1)=O C(=O)(C(=O)C(C)C)N(CC)CC1CCCN1C(c1n[nH]c(C)c1C)=O C1(CNC(C=CC)=O)CCC12CCN(C(C1CC1CC(=O)OC(C)(C)C)=O)CC2 N1(C(COC2CCN(C(=O)C(O)CCn3cncn3)C2)=O)CC(F)(F)C(F)(F)C1 C(=O)(C1=NOC2(CCOC2)C1)OCc1ncn(C)n1 N1(C(C(C)c2cc[nH]n2)=O)CC2CC(C1)N2C(=O)CC1CCCSC1 c1(C(=O)NC2CN(C(c3c(C)nsc3C)=O)CC2O)cccc(Cl)c1[N+](=O)[O-] C(CCF)(C(=O)OC(C)(C)C)NC(=O)NC1C(=C)CC1 Cc1cc(=NCC2CCOC2C)[nH]c(=NCc2cnc(Br)cc2C)[nH]1 C#CC1(NC(=O)C(C)N(C)C(C2CC3CCC2CC3)=O)CCCCCC1 c1(C(=O)NCC2(C)CN(Cc3ccccc3)CCO2)ccc2ncoc2c1 C1(CNC(C2(CNC(CC(C)OC)=O)CC(C)(C)C2)=O)OCCCC1(C)C N1(C(C(CCC)C(C)C)=O)CCC2(CCCN2C(c2cn(C)nc2OC)=O)CC1 N1(C(c2nc(CCOC)oc2C)=O)CC2CN(C(=O)CCCC(C)C)CC2C1 CCC(C)C(C(=O)NCC(CCNC(C1(CCOC)CC1)=O)OC)OC C#CCCCCC(=O)N(C)Cc1ccccc1CNC(=O)C(CC)C(=O)OC C1(CCn2c(C(c3nc(Br)sc3C)NC(CC)C)nnn2)CCC2CC1C2(C)C N1(CC(=O)NCC2CC(O)CN2C(=O)C(O)CC(F)(F)F)Cc2ccccc2C1 c1(C(=O)NC2CCN(C(c3cncc(O)c3Cl)=O)CC2)noc2c1CCCCC2 N1(C(CCCC#C)=O)CC(NC(=O)C(CC)CCc2ccccc2)CC2(CC2)C1 CCC1=NOC(C(=O)NCC(CC2CC2)C(=O)NC23CCC(CC2)C3)C1 N1(C(C(C)O)=O)CCn2ncc(S(C)(=O)=NC(=O)C(C)CS(C)(=O)=O)c2C1 C1(C(N2C(C)(C(=O)NC)CCC2)=O)CCN(C(=O)CC2(OC)CC2)C(C)(C)C1 CC1(C(N2CC(O)(CNC(=O)C3=C(Cl)CCC3)C2)=O)CC(C2CC2)=NO1 c1(C(=O)NC2C(C(C)C)N(C(C3(F)CCOC3)=O)CC2)ccc2nccnc2n1 c1(COC(c2ccc(NCCCC(F)(F)F)cc2)=O)cc(F)cc2nc(S)[nH]c12 CC(C(=O)NOCC(N1CCCC(C(N)=O)C1)=O)N(C)C CCCC(C)(CCC)C(=O)N1CCCOC(CNC(C2OCCC2C)=O)C1 C(CC(C(=O)N(C)C)N1CCC(C(=O)NCc2cccs2)CC1)SC c1(CC(=O)N(C2C3CC(OC)C(C3)C2)C)ccc2c(c1)CCC2 N1(C(C2CC(C)OCC2)=O)CC2(C1)CN(C(c1cnn(C(C)(C)C)c1)=O)C2 O=C1CC(CC(=O)NC(CNC(C2C3CC(F)(F)CC23)=O)C2CC2)CCCN1 C(=O)(C(C)(F)C(C)(C)F)NCCCCC(C)NC(c1cc(C)c(CO)cn1)=O C#Cc1cn(C)nc1C(=O)NC(C(=O)NOCC1CC2C=CC1C2)c1ccco1 c1(C(N2C(C)(CNC(=O)C(O)C(F)(F)F)CCC2)=O)cnn2c1OCCC2 C(CN=c1cc(C(F)F)nc[nH]1)C1CCC(NC(c2ccn(C(F)F)n2)=O)C1 c1(C(=O)NC(C)(C)CNC(c2ccc(Cl)o2)=O)ccc2c(C#N)c[nH]c2c1 c1(C(C)(C)C)cc2c(N(C3CNCC3O)Cc3ccc(CBr)cc3)ncnc2s1 c1(OC)c[nH]c(C(=O)NCC2CN(C(=O)C(C)N(C)C(C)=O)CC2C)cc1=O C=C1CC2(C1)CC(C(=O)N(CC(C)CNC(=O)CC1SC(=N)NC1=O)C)C2 Cc1cc(N)c(C(=O)NC(C2CCCCN2C(=O)CC(F)(F)C(F)F)C)nc1C c1(OCC)cc(N(C)CC2CCN(C(=O)C(C)NC(N)=O)CC2)nc(C)n1 c1(C(=O)NC2CCCN(C(C3CC(CCC)C3)=O)C2C)sc2nnc(S)n2c1C c1(CC(=O)NC2CC(CNC(C3CC3(F)Cl)=O)C2)ccc(O)cc1 c1(OC)ncc(-c2cnoc2)cc1-c1ccoc1 C1(CCCC)CCCCC1N=c1[nH]c2c(c(=NCCc3cc(C)no3)[nH]1)COC2 N1(C(C(C)OCCN(C)C)=O)CCCC2(CNC(=O)CC3CC3)CCCC12 C#Cc1ccc(C(=O)NCC(C(=O)NCCCC(=O)NC)C(C)C)cn1 CC1C(C(=O)NOC2CC2)CCN1C(c1nc(=N)cc[nH]1)=O c1(CC(N2CCC(NC(CCS(C)=O)=O)CC2)=O)ccc(F)cc1F CC(C)CCCC(=O)N1CC(F)CC1CNC(C1CCN(C2CCSC2)CC1)=O C1(NC(C(CC)OC)=O)CCC2(CC1)CC(NC(=O)CCn1cnnn1)C2 n1(CCNC(C(=O)N(C)C)=O)cc(C(C)(C)NC2CC(F)C2)nn1 C12(NC(Cc3c(Cl)cn(C)n3)=O)CCN(C(=O)CC3(C)CCC3)CC1C2 c1(CN(C)C(=O)NCC2CC3CCCCCCC23)nnc2n1CCNC2=O C1(C)(CCC)CCN1C(=O)CCCC1(NC(=O)C(C2CC2)OC)CCC1 N(C1C(=O)Nc2ccc(Br)cc21)C(C(=O)NC(CCC)CC)=O c1(CC(C(=O)NC(CC)CNC(=O)CN(CC)CC)O)ccc(F)cc1 C(=O)(CC(C)C(F)(F)F)NC(CCCNC(CCN1CCN(C(C)C)CC1)=O)C C=CCCC(C(=O)NCC1(C(N)=O)CC1)NC(c1cnn[nH]1)=O N1(C(c2nccs2)=O)CC2(CCN(CC(O)COc3ncc(Cl)cc3Cl)C2)C1 c1(C(=O)NC2(CCCC(=O)NCC3ON=C(C)C3)CCC2)ccc(C#N)c(C)c1 C(C)(C1CCCCC1)=CC(=O)NC1CN(C(c2[nH]c(=NCC)sc2)=O)CC12CC2 c1(C(N(CC(CN(C(=O)Cc2csc(Cl)c2)C)O)C)=O)cc(N)ccc1Cl c1(N(CCC(C)(C)CO)CC)ncc(S(=O)(=O)NCC(C2CCOC2)OC)cc1Cl CC1CCC(CC(=O)NC(CC2CCC2)C(=O)NC2CC(n3cncn3)C2)CC1 N1(C(c2c(C)coc2C2CC2)=O)CCCC(NC(c2c[nH]nc2C(F)F)=O)CC1 C(C(C)C(F)C(=O)N(C)Cc1nccn1CC)NC(CC)=O CC(CC1CCC1)C(=O)NNC(=O)c1cc(-c2ccc([N+](=O)[O-])cc2)[nH]n1 c1(C(=O)OC)ccc(NCc2cn(CCCNC(C3CC(O)C3)=O)nn2)cc1 C(CCCC(=O)N(C)CC1CN(C(=O)C=CC(C)C)CCO1)N(C(C)=O)C C1(C(=O)NCC(C)NC(C(C)SC(C)C)=O)CCCSC1 c1(C(c2nnnn2C2CCCCC2)NCCC(C)(C)C)ccc([N+](=O)[O-])cc1 c1(CNC(COC(CNC(C2C(C(=O)OC)C2)=O)=O)=O)ccc(Cl)nc1 c1(CN2CCC(NC(CC3CC(OC)(OC)C3)=O)C2)cccc([N+](=O)[O-])c1 C1(N(C(C(F)=CCC)=O)C)CCCC2CN(C(c3ccc(Cl)cc3)=O)CC12 c1(C(C(=O)NCCCOCCN(C(C(F)OC)=O)C)N(C)C)ccc(Cl)cc1 n1(CC)nc(C)c(C(N2CCC3C(NC(=O)C4=COCCO4)C23)=O)c1C C(=O)(C(CNC(C1CCC1OC(C)=O)=O)C(C)(C)C)NC(C1(OC)CCC1)C c1(C(N(CC#N)CC#N)=O)[nH]nc2ncc(-c3ccc([N+](=O)[O-])cc3)cc12 C(=O)(C(O)C(C)(C)C)NCC(c1ccc(OC)cc1)NC(=O)CCCC#N C1(F)(CNC(C(c2cccs2)SC)=O)COCCN(C(=O)Cn2ccc(C)n2)C1 CC(C)CCC(F)C(=O)NC(C)CCCCNC(C1CCS(=O)(=O)N1)=O N1(C(CN2C(C)CC2)=O)CCCC1CCNC(c1csc(-c2nc[nH]n2)n1)=O Cc1nc(CO)sc1C(=O)NCCN(CC(C)O)C(=O)CSc1ccccc1 Cc1c(Cl)ccc(C(N2CCCC2C(C)(C)NC(c2ncn(C)n2)=O)=O)c1N Cc1ccc(CSCC(=O)NC2CCOCC2NC(c2coc(CO)c2)=O)cc1 Cc1cccc(-c2ccc(C(N3CC(CO)(NC(C4CC4(F)Cl)=O)C3)=O)n2C)c1 c1(C(=O)NC2C(CC)CN(C(=O)CCCSC)CC2)cnn(C)c1S(N)(=O)=O C(=O)(CC(C)(C)N(C(=O)CC1C=CCC1)C)N(CC(=O)OC)CC c1(C(N2CC(NC(C3(C(C)C)CCC3)=O)C(C)CC2)=O)oc2ccccc2c1Cl c1(C(N2C(CCNC(C3(OC(C)=O)CC3)=O)CCCC2)=O)ccc2n[nH]cc2c1 N1(C(C2CCN(C(=O)OC)CC2)=O)CCC(F)(C(=O)NC2CC(F)C2)CC1 CCCCC(CC)C(=O)NCCOCCNC(=O)CC1CC1C(=O)O.C(CSC)CC C(CCNC(c1scnc1C(C)C)=O)(C(C)C)NC(c1c(OC)scc1)=O n1(CC(N2CC(CNC(C3CC(O)(CC#C)C3)=O)C(C)C2)=O)ncc(C#N)c1N N1(C(c2cncc(OC)n2)=O)CC(O)CCC1C(=O)NC1(C)CCCC1C C1(CC(=O)NCC2CCC(F)(CNC(=O)C=Cc3cocn3)C2)CCS(=O)(=O)C1 N1(C(CC(CCC)CC)=O)CCC2(CCC2)C(NC(=O)CC2C(C)(C)C2(C)C)C1 n1(CCCOC)ccc(=NC(c2nnnn2-c2ccccc2)c2ccoc2)[nH]1 C1(CNC(CS(CC)=O)=O)CC2CCC1N2C(=O)CCc1cnc(C)s1 CC1CC(NC(=O)Cn2nnn(-c3cccs3)c2=O)CN1C(c1coc(Cl)c1)=O CC(C(C)C(=O)NCCOCCOCCNC(C1CC(C(F)F)C1)=O)S(C)(=O)=O C(=O)(C#CC(C)(C)O)NC1CCC(C(=O)NC(C)C(F)F)C1 N(C(=NCCOc1cccnc1)NCC1CCC(C(C)C)O1)Cc1ccc(C)o1 C1(C(=O)NC2(C)CC(NC(Cn3ncc(C)c3)=O)C2)OC2CCC1C2 c1(CC)ccc(Cn2nc(-c3cnn(C)c3)nc2-c2sccc2Cl)cc1 c1(C(=O)NCCCC(C)NC(COCCOC)=O)cc(Br)c(C)s1 C1(C(=O)NCC(C)(O)CN(C)C)(CNC(=O)OC)CCCC1.C1C(=O)N1 c1(C(C(=O)NCCC2N(C(c3cncs3)=O)CCC2)(F)F)ccccc1F c1(C(=O)NC2CC(OCC(=O)NCC(CC)(C)O)C2)cnnc(C)c1 CC(CC(=O)NCC=CCNC(=O)C(C)Oc1ccc(Cl)c(Cl)c1)CC(C)(C)C N1(C(C2(c3ccc(Br)cn3)CC2)=O)CC2CC(CO)(CO2)C1 c1(C(N(C(CCNC(c2c(N)ncc(C)c2)=O)C)C)=O)cccc2c1nnn2C N1(C(C2N(CC)CC2)=O)CCOC2(CCN(C(=O)CC(C)O)C2)C1 c1(C(=O)NC2COCCN(C(=O)C=C3CCOCC3)C2)ccc2c(c1)NCCC2 C(C(C(=O)NCC1(C)CCC1)C(C)(C)C)NC(C(C)OCC(C)C)=O c1(C(=O)NCCc2ccc(CO)cc2)cnn2cccc(-c3ccccc3)c12 C1(OCC)CC2(C1)CC2NC(C1CC1CNC(C1(O)CC1)=O)=O C(=O)(C(O)C1=CCCCC1)N1CCN(C(=O)C2CC2)CC(CO)C1 Cc1c[nH]nc1CNC(=O)CCOCCNC(=O)CSC1CC1 C1(NC(=O)CN(Cc2ccccc2)CC2(CO)CCC2)CCOC2(CCCC2)C1 c1(C(N2C(C)CC(CC(F)(F)F)C2C)=O)cc(F)c2ccccc2c1 c1(C(N(C(CNC(C(C)=NOCC#N)=O)C)C)=O)ccc2cnn(C)c2c1 C1(CC(=O)N(C)CCOCCN(C(=O)COCC(F)F)C)CC12CC2 C1(NC(C)=O)CN(C(=O)CCc2c(F)cccc2Cl)C2CCCCC12 Cn1ncc(C2CC2)c1C(N1CC(CNC(C2COCCO2)=O)C(O)C1)=O CCC(C(C)C)N(C(=O)C(n1cc(CCN(C(C)(C)C)CC)nn1)C)C C(O)(CC(=O)N1CCOCC1C1CC1(F)F)(C(F)(F)F)c1ncc(C)o1 N1(C(Cc2n(C)nnc2)=O)CCN(C(=O)C=Cc2nccs2)C(CC(F)F)C1 C1(NC(=O)C(c2ccccc2)F)CC2(C1)CC2C(N1CC(CF)C1)=O c1(C(=O)NCC(C)CNC(=O)C(C)n2ccnn2)cccc(C(C)(C)C)c1 Cc1ccc(Cl)cc1C(=O)NC(c1cn(-c2cncc(Cl)c2)nn1)C C(=O)(C(C)(C)c1csc(-c2cccs2)n1)NCCN(C)C(C1CCSC1)=O CCC(CC(=O)NC1CC(CO)N(C(C2CC(SC)C2)=O)C1)C1CC1 C1(NC(=O)CNC(=O)C2CC2)CC2CC1CN2C(c1cccnc1O)=O N1(C(C(Cn2ccc(C)n2)C)=O)CCCC(NC(C2CC3(F)CC2C3)=O)C1 CC1CN(C(=O)COCCF)CC1C(=O)NC(C)(C)C(F)F C(=O)(CCCC(C)(C)C)NCCC(CC)(C)NC(=O)CC=CC(C)(C)C CC(C(C)C(=O)NCC1C=CCOC1)NC(=O)CN(C1CCC1)C c1(OC)ccc(Cl)cc1S(=O)(=O)N1CC(F)(F)CC1C(N1CC(O)CC1CO)=O N1(C(c2cc(OC)ncc2Cl)=O)CC2CC3CC2C1C3NC(=O)CNC(=O)OC C1(C(F)F)(NC(C=C(C(=O)NC(=O)C=CCn2ccnn2)F)=O)CCOCC1 C1(NC(=O)C2=CCCO2)CC1C1CCCN(c2ncnc3[nH]ccc23)C1 c1(C(=O)NC2C(C(=O)NCCc3c(Cl)cccc3Cl)C2)cccc2sccc12 C(N=c1[nH]c(=NCC2CCCO2)[nH]c2c1CCC2)c1sc2ccccc2n1 C(CCC(O)C(=O)NCc1ccccc1F)NC(c1c(C)noc1)=O Cc1c(C(=O)NC2CCN(C(=O)CNC(N)=O)CC(C)(C)C2)nn2c1CCCC2 S(=O)(=O)(c1ccc(Cl)cc1Br)N1C(C)C(NC(C)(C)C)CC1 C1(C(N(CCCC)CCCC)=O)CN(C(=O)C(C)CCC)CCC1(C)C N1(C(C2CCCC(NC(C(CC)(C#N)CC)=O)CC2)=O)CC2(C1)CC1(CCC1)C2 c1(C(N(CCCN(C(=O)CSc2ccc(O)cc2)C)C)=O)cnc2sccn12 N1(C(C(F)OC)=O)CC23CCCC2(C1)CN(C(c1cnc(F)c(C)c1)=O)C3 C(=O)(CCC1=CCCCC1)NC1C(NC(C(C2CCCCCC2)C)=O)COCC1 N1(C(c2c(C)nn(C(C)(C)C)c2)=O)CCCC(CO)(NC(=O)CC(C)N(C)C)C1 c1(N2CCC(CCC)(CO)C2)cc(N2CCOC(CC)CC2)nc(CC)n1 C12(CNC(c3c(SC)cccc3F)=O)CN(C(c3cc(F)n[nH]3)=O)CC1CCO2 Cn1cc(C(=O)NC2CC(NC(C3CC(CCO)C3)=O)C2)n(C)c1=O C(C)(C)(CC(=O)NCC1(F)CCC(NC(c2cnc(C)nc2)=O)C1)OC Cc1ccc(Cl)c2[nH]c(C(=O)NC(C)CN(C)C(c3cc(N)ccn3)=O)cc12 C(=O)(C(C(C)CC)N(C)C(c1cnn(CC)c1C)=O)NCC(=O)OCC#C C1(CC)(CNC(=O)C(C(C)C)NC(c2cccc(C)c2)=O)CC(C)(C)C1 N1(C(C(CC)SC)=O)CC(NC(C2C3CCC2(c2ccn(C)n2)C3)=O)CC1C Cc1csc(CC(=O)NCC2CC2CC(=O)NC2(n3ccnn3)CC2)c1 c1(C(=O)NC(CNC(C2(CCOC)CCC2)=O)(C)C)cc(O)c2ccccc2c1 CCC(O)(CN(C)C(c1cn(CCNC(c2ncnn2C)=O)nn1)=O)CC C#Cc1cccc(NC(c2cc(Br)c(C)s2)c2nnnn2CC(=C)C)c1 C(=O)(C(C)(F)C(=O)NC1CC(CCNC(=O)C(C2CCC2)OC)C1)OC c1(C(N2CCCC(NC(c3nc(NC(C)=O)sc3)=O)C2)=O)cc2n(c1)CCCC2 c1(C(=O)NCC(CC)NC(=O)CC2CC(O)C2(C)C)cnc(C2CCC2)cc1C C1(C(=O)NC2(C)CC(NC(C3C(CC)OCCC3)=O)C2)CCCC2(CCC2)O1 CCC(C(=O)OC)C(=O)N1CCCC1(C)C(N1CCC(C(C)OC)CC1)=O N1(C(C(C)NC(C)=O)=O)CCC(NC(c2ccc(F)cc2)=O)C(CO)CC1 C=CCC(CC(=O)NC(C)(CO)CO)NC(=O)CCCNC(C)=O C(=O)(CC1CCCc2ccccc21)N1CC(CNC(C2(C=C)CC2)=O)N(C)CC1 C1(OC)CCn2cc(C(=O)Nc3cc(-c4nn[nH]n4)ccc3Cl)nc2C1 C1(NC(=O)CCN2CCC(F)C2)CCN(C(=O)CCC2CC2)C12CC2 CC(C1CCCCC1)=CCOC(C1(NCC=C)CC1)=O.C1CCCC1 C1(C(N(CC(CNC(C2C(C)C2)=O)(C)C)C)=O)Cc2cc(F)ccc2O1 c1(C(N2CC3CCN(C(CCC(CC)OC)=O)C3C2)=O)ccc2c(c1)C=CCC2 N1(C(C(F)=CC)=O)CCC(NC(c2cccc([N+](=O)[O-])c2N)=O)C2(CCC2)C1 c1(C(=O)NCC2(F)CC(NC(C3CC(OC)C3)=O)C2)cccc2cc(Cl)ccc12 c1(CCC)cc(C(=O)NCCC2(NC(=O)COC)CC2)c(C)o1 N1(C(C(C)NC(=O)NC)=O)CCC2(CC1)CC(NC(=O)C(=O)N(C)C)CO2 C(=O)(C1=NOC2(CCOC2)C1)NCC1(C)CCCN1C(C12CC(F)(C1)C2)=O CC(C1CCCCC1)=CC(=O)NCC(C)(C(C)C)NC(=O)CC1(CO)CC1 CC(N=c1[nH]c(=N)[nH]c(=NCC(C)(F)C(C)(C)F)[nH]1)c1c(F)cccc1Br C1(C(NC(=NCC2CCOC2)NCC2=CCCCC2)C)CCC(F)(F)CC1 c1(SC)cccnc1C(=O)NCC1CCCC(CNC(=O)C(C)SC(C)C)C1 Cc1cnc(CCNC(=O)CCC2CC(NC(C3(C)CCNC3=O)=O)C2)nc1 c1(OC)cc(C)c(C(=O)N(CCCNC(c2c(C)nn(C)c2Cl)=O)C)cc1Cl CCCC(C)(CC)C(=O)N(C)CCN(C)Cc1ncno1 N1(CC)CC(C(=O)N2CC(N(C(=O)C(C)(F)F)C)C(C)(C)C2)c2ccccc21 CC(CC(N)=O)C(=O)NCc1cccc(NC(c2c(O)cncc2F)=O)c1 Nc1cccc(CC(F)C(=O)NC2CC(CO)C2)c1 C1(SC)CN(C(c2cc(Cl)cnn2)=O)CC1NC(=O)C(C)(C)n1cnnn1 C12CCOCC1Cc1cccc(c1)CC2.C(=O)(C(C(C)C)OC(C)=O)NCCC O=S(=O)(c1ccc(-n2cccn2)cc1)NCC(O)C(F)F c1(C(=O)NC(CCNC(Cn2nnc(C)n2)=O)C)cccc2ccnn12 CC#CCCCC(=O)NC(C)C(CO)NC(=O)CCNC(C1CCCO1)=O CCC(C(=O)NC1C2CC3CN(C(=O)Cc4nonc4C)C1C3C2)C(C)(C)CC n1(CC(=O)NCC2(CNC(C(CO)OC)=O)CC2)c(C)ccc1C CCC(F)(F)C(C)(C)C(=O)N1CCC(NC(c2ccsc2C(F)F)=O)C1 c1(C(=O)NCC2CC(NC(c3n(C=C)nnc3)=O)C2)cc(C)cc(C)c1N C1(CC(=O)NCC(CC2CCCC2)C(=O)N2CC3(CC3)C2)CC2(CCC2)C1 Cc1cc(NC(C2CC3CCC2N3C(=O)CC2CCCC23CC3)=O)cc(C)c1C Cc1ncc(-c2cn(C3CCN(C(=O)C#CC(C)C)CC3)nn2)cn1 c1(OC)cccc(C(=O)N(C2CN(C(=O)CC(C)(C)SC)CC2F)C)n1 c1(OCC(N2CC(C(N)=O)C3(C2)CC3)=O)cnc2ccccc2c1 CC1OC2(CNC(=O)CC(C)N(C)C)CC1(NC(c1cccnc1O)=O)C2 N1(C(c2cn(C)nn2)=O)CC(NC(=O)CNC(=O)C(C)(C)C)CC2(CC2)C1 C1(CCC)(NC(c2sccc2C)=O)CCN(C(=O)C(CC)N(C)C)CC1 c1(C2CC(C(=O)NCCNC(C3(C(=O)NC)CC3)=O)C2)ccc(F)cc1 c1(SC)cc(=NC(=O)C2CC(NC(C3(C4(C)CC4)CC3)=O)CCO2)[nH]n1C c1(C(=O)NC2CCCCN(C(C3C(OC)CC3)=O)CC2)cccc(Cl)c1[N+](=O)[O-] C(=O)(C(=O)C(C)CC)N1CC(C(=O)NC(CCCC)COC)C1 CC(C)C(O)CC(=O)N1CCC(CO)C(NC(c2cccc(C(F)F)c2Cl)=O)C1 C1(CNC(C2CCCS2)=O)CCN(C(C2CC2F)=O)C1 N1(C(CC(C)F)=O)CCN(CCNC(C2(C(=O)OC(C)(C)C)CC2)=O)C2(CCC2)C1 S(=O)(=O)(c1c[nH]c(C(N2CCN(C(C3CNC(=O)C(C)(C)C3)=O)CC2)=O)c1)NC Cc1nnc2n1CC(C(N1CC(NC(=O)C=Cc3cscn3)CCC1C)=O)C2 N1(C(c2n(CC#C)ccc2)=O)CCC(C)C(NC(c2cccc(Cl)c2F)=O)C1 CC1(F)CN(C(c2cc(Br)co2)=O)CCN(C(c2cc(Cl)c(Cl)s2)=O)C1 CCCC(C(=O)N1CCOC(C)(CNC(=O)CCCN2CCCC2)C1)S(N)(=O)=O c1(C(=O)NC2CN(C(CCC(=C)Cl)=O)CC2O)cc2cccc(C)c2s1 c1(C(=O)NCC2CC(OC)CN2C(c2ccnc(O)c2)=O)ccn2ccnc2n1 Cc1ccc(C)c(C(=O)NC2CCC(NC(=O)NC3CCC3)CC2)c1C Cc1cc(C(=O)NC(C)CN(C)C(C2(C)CCNC(=O)C2)=O)cc(C)n1 c1(NC(COCC)COC)[nH]c(=NCCNS(=O)(=O)C2CC2)nc2scnc12 Cc1oc(C(=O)NCC2CN(C(=O)C(n3cc(Cl)cn3)C)C2)cc1CO C1(O)(CN(C)C(C2CC(N(C)C)C2)=O)CCN(C(=O)C(C)(C)CCF)CC1 C1(C(=O)N(CC(C)C(=O)N(CC(O)CF)C)C)(CC)CC(C)(C)C1 CC1Cn2nccc2CN1CCN(CCc1cccc(F)c1)CCN c1(CC(N2C3C(CNC(C4CCS(=O)(=O)C4)=O)C(C3)C2)=O)cc(F)c(F)cc1F C1(O)(CCNC(CCOC(C)C)=O)CCN(C(=O)C(C2CCCCC2)C)C1 S(=O)(=O)(c1ccc(NC(c2cnn(CCOC)c2)C)c(F)c1)N1CC(COC)C1 N1(C(c2sccc2Cl)C(=O)NCCCF)CCCCC(N2CCCC2)C1 CCC(O)CC(=O)NC1CCCN(C(=O)Cc2ccc(OC)cc2)C1 C(CCCCCC(=O)N1CCC(NC(C2C=CCC2)=O)C12CCC2)SC C#CCC(C)(C)C(=O)NCC12CC1CN(C(c1c(C)nn(C)c1Br)=O)C2 C1(CNC(C2CC(SC)C2)=O)CN(C(c2ccc(N)cc2O)=O)CC12CCC2 c1(C(N2C(CCNC(CCN(C)CC)=O)CSCC2)=O)ccn2cccc2c1 C(C(CO)N=c1[nH]nc(C(C)C)o1)NC(c1cc(CC)n(-c2ccccc2)n1)=O C1(NC(c2ccc(C(F)(F)F)o2)=O)CCC12CN(C(=O)CCC1CCOCC1)C2 N1(CC=C)CCC(C(N)=O)CC1.C1(=O)CCC(=O)N2CCCC(C2)CN1C Cc1cc(CNC(=O)NCC2CCS(=O)(=O)N2C)nc(Cl)c1Br c1(CN(C2CN(C(c3cc(C)nn3C(F)F)=O)C2)C)cc(F)cc(Br)c1 C#CC1CN(C(C2C=CCC2)=O)CCN1C(c1cc(O)ccc1C)=O C1(OC)CCn2cc(C(=O)NCCC(C)NC(c3c[nH]nc3C(C)C)=O)nc2C1 c1(CC)cc(Br)c(C)cn1.C1(CSCC)CNCCS1 C(=O)(C(COC)C(F)(F)F)N1CCCCC(NC(c2ccc(CC)s2)=O)C1 c1(C(=O)NCC(CC)NC(CC(=C=C)C)=O)ccc(-c2ccccc2)cc1C C(=O)(C(C(F)(F)F)C(F)(F)F)N1C(CN(C(C(CCCC)C)=O)CC)CCC1 N1(C(c2cnc(SC)nc2O)=O)CCC2C(C1)CN2C(=O)C1=CC(C)(C)C1 N1(C(C(CCOC)NC(=O)C(C)=CC(C)(C)C)=O)CCCNC(=O)C1C N#Cc1ccnnc1NC1CC(CCNC(C2CCCO2)=O)C1 Cc1c(F)cc(C(=O)NCC(CNC(c2cc[nH]n2)=O)CO)c(F)c1N C12(NC(CCc3c(C)noc3Cl)=O)CCCN(C(=O)C(C)(C)O)CC1C2 Cc1nc(C(C)C)oc1C(=O)NCCCN(C(=O)Cn1nnc(C2CC2)n1)C N1(C(c2c(C)snn2)=O)CCCN(C(=O)Cc2ccc(C(C)C)cc2)CC1CO C12(C(=O)NC3C(CCC)CN(C(C4COCCC4C)=O)C3)CCC(C1)OC2C N1(C(c2c(-c3cc(=NC)[nH]cc3)cncn2)=O)CCOC2CCCC12 N1(C(c2c(C(=O)OC)c(C)on2)=O)CCC(NC(c2cc(C)nn2C)=O)C(C)C1 N1(C(c2cccc(CC)c2)=O)CC(N=[N+]=[N-])CC1C(=O)NCC(O)CC(C)(C)C N1(C(C=CCC)=O)CCOC(C(C)NC(=O)CCCn2c(O)nnc2O)C1 C1(C)(NC(c2cnc(C)o2)=O)CCN(C(c2cccc(CCO)c2)=O)CC1 c1(CC)[nH]nc(C(=O)NCC=CCNC(c2nnn(C(C)C)c2C)=O)c1Br C1(C#N)(C(=O)NCCCCC(N2CC=C(C)CC2)=O)CC2CC2C1 C(C(CC(C)C)C(=O)N1CCC(OCCNC(=O)C=CCOC)C1)OC c1(C(=O)NCC2(C)CCN(CCn3c(C)ncc3)CC2)coc2c1C(=O)NCC2 N1(C(CCNC(=O)OCC)=O)CC(NC(C2CC(O)CN2C(C)=O)=O)C(C)C1 c1(C(=O)NC2CC(NC(COCCCN(C)C)=O)C2)ncnn1C N1(C(C2CCC(C)CN2C(C2CCNC2=O)=O)=O)CC(C#N)C2(CCC2)C1 c1(CC)ccccc1CC(=O)NCC12CC1CN(C(c1ocnc1C)=O)C2 N1(C(c2cccc(C)c2N)=O)CC2CC(C)N(C(=O)CC3CCC(C)(C)C3)C2C1 N1(C(c2ccnnc2)=O)CCC2CC2(C(=O)N(C2CC2)CC2CC2)CC1 C(=O)(C#CC(C)(C)O)NCC1C(C(N2CCCC(OCCC)C2)=O)C1 CC1CN(c2ccccc2CNC(c2[nH]nnc2Cc2nn[nH]n2)=O)CC(C)O1 c1(CC(=O)NC2(C)CN(C(C(COC)O)=O)C2)noc2cc(F)ccc12 O=C1CCC(C(N2CCC(NC(=O)C(C3(O)CCCC3)F)CC2)=O)CN1 C(=O)(C(CO)C(F)(F)F)NC1(C2CN(C(C(c3ccc(C)s3)C)=O)C2)CC1 C1(C(N2CC(CNC(CNC(CCC)=O)=O)C(O)C2)=O)CC(=O)NC(=O)N1 C(CCN(C)C(C1CCCC1)=O)(C(C)C)NC(C1(OCC)CCOC1)=O Cc1cccc2[nH]c(C(N3CCCCC3CNC(c3cccc(O)n3)=O)=O)cc12 Cc1ccccc1C=CC(N1CC2(NC(c3cc(C)c(C)[nH]3)=O)CCC1C2)=O N1(C(CSCC)=O)CCC2(CNC(=O)C=Cc3ccccc3)CCCCC12 O=C(C#Cc1ccccc1)N1CC2CCCN(C(c3ccnc(Br)c3)=O)C2C1 CC(CC(=O)NCC(CO)NC(=O)C(c1ccc(Cl)cc1)O)C(F)(F)F c1(CC(=O)NC(C)C(=O)NCC2CCCCS2)ccc(O)nc1 N1(C(CC2(OCC)CCC2)=O)CC2CN(C(C3COCCC3(F)F)=O)CCC12 N1(C(Cn2ccc(=N)[nH]2)=O)CCC(NC(c2cc(C3(C)CC3)n[nH]2)=O)C(CO)C1 c1(-c2n(CCOC)ccn2)ncc(-c2ccc(N)cc2C2CC2)cc1F N1(C(=O)Cc2cnccn2)CC2CCC1CN2C(=O)C=C1CCCCCC1(F)F CC1CC(NC(c2cnc(Cl)c(N)c2)=O)CN(C(c2ccc(C3CC3)s2)=O)C1 c1(C(=O)NC2CN(C(c3cnn(C)c3N)=O)CC2(C)C)coc2c1C(=O)NCC2 CC1CCc2onc(C(=O)NC3(C)CN(C(c4ccnc(Cl)c4N)=O)C3)c2C1 N(C1CCOc2c(OC)cc(C)cc21)C(N(C1C(OC)CCOC1)C)=O C(=O)(CC(C)(C)C)NCC(N1C(C(C)NC(C2COC(=O)N2)=O)CCC1)=O c12ncc(cn1)C(=O)NC2.C1(CCCOC)(CNC(=O)CC(C)C)CCCC1 C(C1=CCN(C(=O)C=Cc2ccc[nH]2)CC1)NC(Cn1c(C)csc1=O)=O N1(C(CNC(CC(C)(C)C)=O)=O)CCC2CN(C(c3ccns3)=O)CC12 C(C1=NOC2CN(C(c3cn(C4CC4)nn3)=O)CC12)NC(c1cc(C)c(C)[nH]1)=O C1(C(=O)OCC)CCCC(NC(c2cnn(C)n2)(C)C)C1 C1(NC(c2c(CC)cccn2)=O)CCN(C(C23CCOC(C)(C2)C3)=O)CC1C S(=O)(=O)(c1ccc(I)cc1[N+](=O)[O-])NCCc1cc(C(C)(C)C)on1 C1(CN(C(=O)CC2(C)CC(F)(F)C2)C)CN(C(=O)C(F)C(F)(F)F)CC12CC2 C(c1ccc(F)cc1)=C(C)C(=O)NC1CC1NC(=O)CCc1cnc(O)[nH]1 c1(C(=O)NC2CC3(CN(C(Cn4c(C)nnn4)=O)C3)C2)c[nH]c(=O)c2ccnn12 Cc1nn(C)c(C(=O)NC2CCC2CNC(=O)C(F)(F)C2CCCC2)c1[N+](=O)[O-] C1(O)(C(C)NC(=O)COC(F)F)CCN(C(c2cnn(C3CC3)c2)=O)C1 CC(CC(F)F)C(=O)N1CCN(C(C)CNC(=O)CSc2ccncc2)CC1 CC1(C)CC(CNC(=O)N(CCO)CC2CCCN(C3CCC3)C2)c2ccccc2O1 C(c1cccc(F)c1)=CC(=O)NC1CC(C(N2CCCC(N(C)C)C2)=O)C1 N1(Cc2c(C)nc(C)s2)CCC(C)C(NC(=O)CCC2NC(=O)NC2=O)C1 c1(NC(C2COCCN(C(CSC)C)C2)=O)[nH]nc2ncccc12.C(CCS)N Cc1cncc(C(=O)NCCN2CCN(Cc3nc(Cl)nc(C)c3Cl)CC2)c1Cl c1(CC)n[nH]cc1C(c1nnnn1CC1CCCO1)NCCC1(SC)CCC1 CC(C(=O)Nc1ccccc1F)(C(F)(F)F)NC(=O)CN1CC2CC=CCC2C1 CC(O)C(C)C(=O)NCCN(C1CCCC1)C(=O)COCc1ccccc1F CC(C)(C)C(O)C(=O)N1CC(NC(C2CCCC(=O)C2)=O)C(C)(C)C1 c1(C(=O)NCC2(F)CCC(NC(CCOCC#C)=O)C2)cc(C)c(F)cc1N c1(CCNC(c2cnc(OC(C)C)nc2C(F)(F)F)=O)ccc2c(c1)CC(C)O2 CCCCS(=O)(=O)CC(=O)NC1CC(NC(C2CC(O)(C(F)F)C2)=O)C12CCC2 C(=O)(C(C)CC(C)CC(C)C)NCCN(CCC)C(C1OCCC1CC)=O N1(C(c2cnc(SC)s2)=O)CCN(C(c2ccon2)=O)C(CC(F)F)C1 N1(CC(=O)N(C2CC2)CC2N(C(C=C(C)Cl)=O)CCC2)CCC(F)(F)C1 N1(C(C(C)O)=O)CCC(NC(c2cc(Cl)ns2)=O)C1C1CC1 C1(NC(c2cc(COC)on2)=O)CC(O)CN(C(=O)CCc2cccc(Cl)c2)C1 C1(C(=O)NCC(C)NC(=O)C(C)(C)c2cncnc2)CC(C)(C)CO1 CC(C(=O)NCCC1(CNC(=O)C(C2CCCO2)C2CC2)CC1)N(C)C c1(C(N(CC(C)C(=O)NC(C)Cc2ccco2)C)=O)c[nH]c2ncccc12 Cc1ccc(C(C)C(N2CCCC2C2CCCOC2)=O)o1 CCC(C)C(O)C(=O)N1CCN(C(c2cc(C(N)=O)cc(F)c2)=O)CC1C(C)C C#Cc1cnn(C)c1C(=O)NC1CCCN(CC(F)(F)F)C1=O NC(Cc1ccccc1)C(=O)NCCC1CCC1 C=CC1(O)CCN(C(=O)C(N)CC2CCOC2)C1 CC(C)(C)CCC(F)C(=O)NC12CCCC1N(C(=O)CS(C)(=O)=O)CC2 C(CCS(C)(=O)=O)CN1CCC(C(C)NC(=O)OCc2cnn(C)c2)C1 C(=O)(CS(=O)(=O)C12CC(C1)C2)N1C2CC(NC(C3CC(=C)C3)=O)CC1CC2 N1(c2ccc(NC(=O)NC3(c4cccc(C)c4)CC3(F)F)cc2)CCS(=O)(=O)CC1 C1(NC(CNC(C2CCCC2)CC)=O)CCOCC1 n1(CCCC)nnnc1C1(NC2(CSC)CCCC2)CCC1CCOC CN1C(=O)OCC12CN(C(=O)CC(F)(F)c1ccncc1Br)C2 c1(CN(C)C(=O)OC(C)(C)C)ncc(C(=O)NCC23COC(C2)C3)cn1 S(=O)(=O)(c1cnc(NCC2(Cl)CC2(F)F)c(Cl)c1)NCC(C)N(C)C C1(C(=O)NC2(C(C)C)CC2)CCCCN1C(=O)CC1CCCC(C)C1 c1(C(=O)NC(CCOC)CNC(=O)C=Cc2cnccn2)cc(F)cc(N)c1F c1(CNC(C(C2CCN(C(CCSC)=O)C2)C)=O)c(Br)cnn1C Nc1c(C(N2CCC3(COC(COc4ccccc4)C3)C2)=O)cc(F)c(F)c1F C1(C)(C(C)C)C(=O)N(C)C(C)CN1.CN=c1[nH]cc(C(=O)OC(C)(C)C)s1 C12(NC(c3c(C)ccnc3Cl)=O)CCCC1CN(C(=O)COc1ccccn1)C2 N1(C(C(C)CC2CC2)=O)CCCC(N(C)C(C2(Br)CC2)=O)C1 C(CC(C)C)(C(=O)NCC(=O)N(C)O)N(C(CCN(C)CC)=O)C Cc1ccc(C(=O)NCC2C3CN(C(c4n[nH]cc4Cl)=O)CC23)c(=O)n1C Cc1cc(Br)c(Cl)cc1NC(C1CC(F)CN1C(C1CCCN1C)=O)=O C=CCCN=C(NCC(N1CCOCC1)C)NCC(O)C1(C)CC1 c1(OC)cccc2c(C(N3CCC(C)C3CNC(=O)CCC(C)(F)F)=O)coc12 C1(CNC(C2CC(C)(CC)C2)=O)CN(C(c2c(C)cnn2C)=O)CC2(CCC2)O1 N#CC1CC2(CC(NC(C3CC(NC(=O)C(O)CC(N)=O)C34CCC4)=O)C2)C1 c1(C(=O)NC2CN(C(CSC(C)C)=O)C3C2C3)cnc2cnn(C)c2c1 C#CCCC(C(=O)NCC(C1CCCCC1)O)NC(=O)C(n1cc(C)cn1)C CCC(CC)C(C(=O)NCCCC1CCCN1C(c1ccco1)=O)OC N1(C(COCc2cc(C)no2)=O)CCC(NC(=O)C2=CCCS2)C(CO)C1 c1(C2N(C(c3csc(C(F)(F)F)n3)=O)CCC2)cncc(Cl)c1 Cc1cccc2c1OC(C(N1CCCC(NC(=O)Cn3cc(C)cn3)C1C)=O)C2 N1(C(c2c(OC)cncn2)=O)CC2CCC1CN2C(C1CC2(C1)CC(C)C2)=O c1(C(C)NC(C2(C(C)NC(=O)C(F)C3CCC3)CC2)=O)ccccn1 C(=O)(CCCC(C)(C)C#N)NCC#CC(=O)NCc1cc(C)oc1 c1(C(=O)NCC(CC(F)(F)F)NC(c2cc(F)c[nH]2)=O)cccn2nccc12 N1(C(C=C(C)C(F)F)=O)CC(F)(F)CC1CCNC(=O)COC(F)F c1(C(N2CCN(C(C(COC)C)=O)C(C)CC2)=O)cc(OC)cc2c1OCC2 C1(NC(c2snc(Cl)c2Cl)=O)CCCC(NC(c2cnn3c2CCC3)=O)CC1 CCC(CC(=O)NCC=CCNC(=O)C(CC)OC)c1ccc(OC)cc1 c1(C(N2CCC(C(C)NC(C(CC)F)=O)C2)=O)cc(N)ccc1O CC(CC(=O)NCC1COC(CNC(=O)Cn2nc(O)ccc2=O)C1)P(C)(C)=O CC1(C)CCCC(CC(N2CC3CC3(NC(=O)Cc3ccsc3)C2)=O)C1 c1(CNC(=O)NC2CCN(C(=O)OC)C2)cccc(CN=[N+]=[N-])c1 c1(NC(C2N(C(CCCN(C)C)=O)CC2)=O)c(C#N)cnn1C(C)(C)C N1(C(CC23C(CN(C(CC(CC)(C)C)=O)C2)CC3)=O)CC2CC=CCC2C1 N1(C(C2=CCC(NC(CC3CC(SC)C3)=O)C2)=O)CCC12CCC(C)CC2 CCC(C)C(O)C(=O)N1CCOC(CNC(=O)CSCc2csc(=N)[nH]2)C1 Cc1ccc(OCC(N2CCCC2(C)CNC(=O)CN2CCC2C)=O)c(C)c1 C1(C(=O)NCC(c2ccccc2)CNC(C2(CF)CC2)=O)CC2(C1)CC2F C(=O)(C(CCC1(C(C)(C)OC)CC1)C(C)C)NC(C1CC(O)C(F)C1)=O C1(C(=O)NCC(CNC(c2cnc(CCCC)s2)=O)CO)CC12CCOCC2 Cc1nc2sccn2c1C(N1CCC(NC(C2CC3CCC(C2)C3O)=O)C1C)=O c1(C(=O)OC)ccc2c(n1)CCCN2C(c1cc2ccccc2nc1Cl)=O N1(C(C(N2CCOCC2)C)=O)CCC2(CCCC2NC(C2C(C)(C)C2(C)C)=O)CC1 N1(C(C(C)NC)=O)CCC2(CCCC2C(=O)N(c2ccc(-n3cccn3)nc2)C)C1 N1(S(CCCC)(=O)=O)CCC2(CC(C(=O)Nc3cc(C(F)F)c(Cl)cc3F)=NO2)C1 C1(OC(c2ccc(S(=O)(=O)N3CCCC3)o2)=O)CCc2ccccc2C1 c1(OC)nc(C)ccc1C(N1CC2(CCN2C(c2cc(Cl)cnc2Br)=O)C1)=O O(NC(=O)C(C1(O)CCC1)NC(=O)CC(C)(C)SC)CC#C Cc1cc(=NCCC2CCC23CCC3)[nH]cc1S(=O)(=O)N(C)CC1(N(C)C)CCCC1 N1(C(CN(C)C)=O)CCN(C)CC1C(N1CC(O)C(O)C1)=O CC1CCCC1NC(=O)NCCN(C)CC1CCOCC1 C1(C)(C(=O)NC(c2ncc(C)o2)C)CCN(C(c2nnn(C)c2C)=O)C1 C1(O)(CCNC(Cc2c(C)ccnc2)=O)CCCN(C(C2CC2C(F)F)=O)C1 C1(NC(c2ccc(CCC)cc2)=O)CN(C(=O)C(O)CC)CC2(CCC2)C1 c1(C(=O)NCCOCCNC(C(CCSC)O)=O)ccc(OC)c2ccnn12 c1(C(C)(CC2CCOC2)OCCO)nnnn1C1CCC1.n1(NCCC)ccnn1 c1(CC(=O)N(CCCNC(c2sccc2C)=O)CC)cc(Cl)cnc1C CCC(CC(=O)NC(c1ccoc1)C)NC(c1ccccc1NC)=O C1(OCC)CN(C(C2(C(C)C)CC2)=O)CC1CNC(=O)C=CC(C)(C)SC c1(C(N2CCN(C(Cc3cccc(CC)c3)=O)CC2C)=O)cnc2c(c1)NCC2 N1(C(C2C(C)(C)C2)=O)CCC2CCN(C(C3(C)CC(F)C3)=O)CC2C1 C(CCC(N)=O)(C(=O)N(C1CCC1)C(C)=O)OC(CC1CC(NC)C1)=O CCCCC(C(=O)N1CCC2(CC=CCO2)C1)C(C)C c1(C(=O)NCC2(NC(CCCSC)=O)CCCCCC2)c(C)cc(O)nc1C C(C(O)(CNC(=O)CCC1(C)CN(C(=O)C(c2ccnn2C)O)C1)CO)OC c1(OC)cccc(C(=O)N(C)CC2(O)CCCN(C(c3conc3C)=O)C2)c1F C(=O)(C1CCCc2sccc21)NC1CN(C(c2c(C)cc(C)s2)=O)CC1C C1(CNC(=O)CC=C(Cl)Cl)CCCC2(CN(C(=O)C=CC3CCCCC3)C2)O1 C1(C(=O)NCC2(F)CN(C(=O)COCCN(C)C)C2)SC2C=CC1CC2 N1(CC(N2CC(SC)C(NC(c3ccc(C(C)C)o3)=O)C2)=O)C(=O)CN(C)C1=O N1(C(CCOC)=O)CCC(NC(=O)Cc2ccccc2S(C)=O)CC(C)(C)C1 Cc1nn2cc(-c3nc(C(C)CCCC(F)(F)F)no3)cnc2c1Br c1(C(N2CC3C(NC(c4cccc(O)n4)=O)(C3)C2)=O)cc(F)cc2nc(S)[nH]c12 C1(CNC(COCC(C)(C)C)=O)(NC(c2ccc(O)c(Cl)n2)=O)CCCCCC1 C1(O)(CNC(C(C)(F)F)=O)CCCN(C(=O)CN2CCC(C(N)=O)CC2)C1 c1(C(=O)NCCOCCN(C)C(C2CCC(O)C2)=O)cccc(C(F)(F)F)c1 CC(C)C(C)CC(=O)NCCCCN(C(=O)COCCCN=[N+]=[N-])C c1(C(N2CCC(NC(CN(C(C)C)C)=O)C2C)=O)noc2c1CC(C)CC2 c1(OC)cc(F)c(Br)cc1C(=O)NC1CC1NC(C1CCCCC1(F)F)=O C(=O)(C(C(C)(C)C)OC)NCCC1(C(=O)NC(C=C)CO)CCOCC1 N1(C(C(COC)OC)=O)CCC2(CC1)CC2(CO)CNC(=O)C1=CCCC1 C(=O)(C(C(C)(C)C)OC)NCC(CCOC)NC(c1cscc1OC)=O C1(CC(C(=O)NCC=C)N(C)Cc2nc[nH]n2)CCC(F)(F)CC1 Cc1sc2ncc(C(N3CC4CCC3CN4C(c3cc(Cl)ccn3)=O)=O)n2c1C c1(C(=O)NCCCC2CCCN2C(C2CCCS2(=O)=O)=O)ncn2c1CCCC2 CC(C)CC(C)C(=O)N(C1CCCC1)CCNC(=O)CC(C)(C)Cc1ccccc1 C(=O)(CCP(C)(C)=O)N1CCC(O)(C(C)NC(CSCC#C)=O)C1 C1(C(=O)NCC2(CNC(c3cccc(F)c3)=O)CC2(F)F)CCn2cncc2C1 c1(C(CNC(c2n(CC)nnc2)=O)NC(c2ccnnc2)=O)ccc(C)cc1 C1(NC(N2C(C(C)(C)O)CCC2)=O)CCCCC(F)(F)C1 C(C(CC)(CC)CO)NC(c1c(CNC(CCC)=O)n[nH]c1)=O Cc1cc(C2CC2NC(C2CC(c3ccc(F)c(F)c3)(C(=O)O)C2)=O)ccc1Br c1(C(=O)NCC2(F)CC(NC(c3cc(CC)ncn3)=O)C2)ccnc2cc[nH]c12 c1(C(=O)NC23CCCC2N(C(=O)Cc2cc[nH]n2)CC3)ccc2oc(O)nc2n1 C1(N(C(COCc2ncc(C)o2)=O)C)CC2CCC(C1)N2C(C1CCC2CC12)=O N1(C(c2c(C(C)C)[nH]cc2)=O)CCC(CF)(NC(c2ncccc2F)=O)C1 c1(COC)nc(C)c(C(=O)NC2CCC(Cn3cc(-c4cnn(C)c4C)nn3)C2)s1 c1(C(=O)NCCOCCCN(C(CCC=C=C)=O)C)ccc(C(C)=O)c(C)c1 c1(C(N(CCCCN(C(C2N(CC)CC2)=O)C)C)=O)nn(C)cc1Cl N1(C(CS(=O)(=O)NC)=O)CCC2(CCCCC2NC(c2cccs2)=O)C1 C1(C(=O)NC(c2nncs2)C)CCCN(C(C2CNC(=O)N2)=O)CC1 C1(NC(C(C=C)(C)CC)=O)CCN(CCCC2CCCCO2)CC1(C)C C1(c2ccccc2)(C(N2CC(C)(NC(C3CCC(C)S3)=O)C2)=O)CC2(CC2)C1 C1(C2CCCO2)(CNC(CC)CNC(=O)C(F)CC2CCOCC2)CCOCC1 N1(C(c2cc(CCC)on2)=O)CCC(CC)(NC(c2ccoc2Br)=O)CC1 c1(NCCC(=O)Sc2n(CC)c(-c3ccccc3C)nn2)cc(F)cc(F)c1 N1(C(C2(OC)CCCOC2)=O)CC(O)(C2CCN(C(=O)CSC3CC3)CC2)C1 C(=O)(C=C1SCC(=O)N1C)N1C(CNC(C(C)C2CCOC2)=O)CCCC1 N1(C(CCC=C)=O)CC2CCC2(NC(c2ccc(-c3csc(=N)[nH]3)cc2)=O)C1 N1(C(C(C)CC2CCC2)C(=O)NCC2CC2)CCc2c(O)cccc2C1 C(=O)(C1SCCc2ccccc21)NCCC1(O)CN(C(C(C(C)C)CO)=O)C1 c1(CC)nccnc1C(=O)OC.C1(CN2C3CC3C2=O)OCCO1 N1(c2cc(C)c(C3CC3)c(C)n2)CCC2(CC1)CC=CC(=O)N2C c1(C(=O)NC2C(NC(c3csc(CO)n3)=O)COC2)csc(Cl)c1Cl n1(CCC)nnnc1C(C)(COC(C)C)NC(C)COC Cc1cccc(C(N2CCCC(N(C)C(c3cc(C)n(C)n3)=O)CC2)=O)c1F N1(Cc2ccc(OCC)nc2C)CCc2cc(OC)c(OC)cc2CC1 c1(CC)c(C(=O)NC2CC2NC(c2cc(OC)c(Br)s2)=O)cnn1CC C1(CCOC)CN(C(=O)C(F)(F)C2CCCC2)CCN1C(c1csc(Cl)n1)=O c1(NC)snc(C)c1C(=O)NCCCCCCNC(C1CCCC1(C)C)=O O=C(O)CC(C1CC(F)(F)C1)NC(=O)NCC1CCC(c2ccccc2)C1 C(CC(C(=O)NC(c1nncn1C)C)NC(=O)CCc1nc(O)n[nH]1)SC C1(NC(C2N(C(C)=O)CCCC2)=O)CC2(CCN(C(c3cc(CN)no3)=O)C2)C1 N1(C(C(c2ccccc2)NC(C)=O)=O)C2CCC1CN(C(c1ccccn1)=O)CC2 C1(C)(C(N2CC(NC(CC3C(C)C3(F)F)=O)C2)=O)CC(C(C)(C)C)=NO1 Cc1ccc(F)c(NC(C2CCC(CNC(=O)CCC3CCCN3C)CC2)=O)c1 CC1(C)CC(C)(CNC(C2CCCCS2(=O)=O)=O)CN1C(c1csc(C#N)c1)=O C1(NC(C2CCC(=C)CC2)=O)C2CCC(C2)C1C(=O)NOCC(C)C O(C=C(C#N)C(=O)N1CCN(C(=O)C(c2ccc(C)s2)C)CC1C)CC N1(C(C(C(C)C)N(C)C)=O)CCC2CCN(C(c3cccs3)=O)C2C1 c1(C(=O)NC(C)C(C)NC(C2CC(N(C)C)C2)=O)ccccn1 C=Cn1nccc1C(=O)N(CC(O)CNC(c1cc(O)nn1C)=O)C Cc1ccccc1C=CC(N1CC2(C(=O)NC3CCCC3CO)CC1CO2)=O Cc1ncc(C(=O)NCC(C)CNC(=O)C(C)N(C)Cc2ccccc2)c(C)n1 c1(C(=O)NC(CC#C)C(=O)NCC2(O)CN(C)C2)cc(C)c(N)cn1 N1(C(C(c2cccs2)NC(COCC)=O)=O)CCC1(C)CC C(CCC(C)C)(C(=O)NC1CC(N(C)C(c2cc(C)cs2)=O)C1)NC(=O)OC C1(C(=O)NC2(CF)CN(C(CC3CCC(C)(C)O3)=O)C2)CC2C=CC1C21CC1 C(=O)(C(COC)CC(C)C)N1CC2(N(C(C(C)SCCCC)=O)CC2)C1 CC(C)CC(F)(F)C(=O)NC(C1CCN(C(=O)COCc2ccccc2)C1)C C1(C(=O)NC(CC)(C)CCNC(c2ccnnc2)=O)CCc2cnnn2C1 C(=O)(C1=CNC2=NCCC2=C1)N1CCCC(C(C)NC(Cc2nnc(C)o2)=O)C1 c1(C(=O)NC23CC(CNC(C4CC(C)C4)=O)(C2)C3)cc(N)c(F)c(F)c1Cl C1(NC(Cc2cccc(C)c2F)=O)CN(C(C2CC3(CC3)C2)=O)CC(F)(F)C1 C1(NC(C2N(C(COC3(C)CCCC3)=O)CCC2)=O)CCOC12CCCC2 N1(C(CC(C)OC)=O)CCCC(C)(NC(c2cccc(-n3cnnn3)c2)=O)C1 c1(C(c2n(CCC)nnn2)NCC(C)(C)CCO)cc2cc(Cl)cnc2o1 C12(C(N3C(COC)CC3)=O)CCCC1CCN2C(C1(O)CCCC1)=O N1(C(=O)CCC2CCC2)CCN(C(c2noc3c2CCCC3)=O)CC(O)C1 C(=O)(CCC(F)(F)CN=[N+]=[N-])NCC1N(C(c2c(C)cc(=O)n(C)n2)=O)CC=C1 Cc1ccc(N(C)C(C2CCN(c3nccc(Br)n3)CC2)=O)c(C)c1 c1(C(=O)NC(CNC(c2c(C)coc2C)=O)(C)C2CCC2)ccc2c(c1)OCC2 c1(C(=O)NCC2C=CC(NC(C(C)NC(COC)=O)=O)C2)n[nH]c(C)c1Cl C1(CC(N2CC(CC(C)NC(C3(C(=O)NC)CCC3)=O)C2)=O)CCCC(C)C1 c1(NC(C)=O)cc(C(=O)NC2CC3(C2)CC32CCC2)ccc1[N+](=O)[O-] C1(CNC(c2ncccc2Cl)=O)C2CCC1CN(C(=O)Cn1ccccc1=O)C2 C12(NC(c3snc(C)c3Br)=O)CCCC1N(C(=O)C1CC1)CCC2 c1(C(=O)NC(C=CC(=O)Nc2c(C)cc(F)nc2)C)coc2ccccc12 c1(C(N2CC(NC(C(C)CC3CCC3)=O)C(C)(C)C2)=O)c(F)cc(N)cc1F N1(C(CC(=O)NCC)=O)CCCC(C2CCCN(C(=O)Cc3cnc[nH]3)C2)C1 N1(C(c2ccc3nccn3c2)=O)CCC2CCN(C(=O)Cn3cc(Cl)cn3)C2C1 Cc1c(C(=O)NCC(C)N(C(=O)CCn2ccnc2)C)c(-c2cccs2)cn1C c1(CNC2C(C(=O)NC3CCNC3=O)C2)c(F)cc(F)cc1F N12CCCC(C)(C1)CC2.n1(C(C)C)ccc(C(=O)NC2CCOC2)n1 N1(C(C(Cc2cc[nH]n2)NC(c2c(NC)cccc2)=O)=O)CCCCCCCC1 c1(C(c2nnnn2C(C)C)NCCOC(COC)=O)ncc(CSC)s1 c1(NCC2C(NC(C3(O)CCC(C(C)CC)CC3)=O)C2)cc2ccc(C)cc2[nH]1 C1(C(N(CC(C)NC(=O)COCC(F)F)C)=O)COc2ccc(Cl)cc2C1 N1(C(CCCOCC)=O)CCN(C(=O)C(C)Oc2ccc(Cl)cc2)CC1C c1(N2CC=C(C)C2)nc(N2CCN(c3nc(Br)cs3)CC2)nc2scnc12 c1(CCNC(C2CN(C(=O)CC3CC3)CC2(F)F)=O)c(F)cccc1Cl c1(NCC2N(C(C3(CC(=O)OCC)CC3)=O)CCCC2C)cc(C)c(C#N)cn1 C1(NC(c2c(C)nns2)=O)CCN(C(C2CCC3CC3CC2)=O)CC1(C)C C1(C(=O)NCC2(CCNC(C3(C)CCC4CC4C3)=O)CC2)CN=C2N=CNN2C1 C1(NC(C(C)OCC#C)=O)COC2(CCN(C(=O)CCc3cncnc3)CC2)C1 C12(C(=O)NCC(C)(C3CC3)NC(=O)C=CCO)CC(F)C1C2 CC(c1ccc(F)cc1)=CC(=O)NCC1CN(C(=O)Cc2n[nH]c(C)n2)CC1C C1(CNC(C(C)SCCCC)=O)CN(C)CCN1C(c1cc2[nH]ccc2s1)=O c1(C(N(c2ncccc2N)C)=O)cccc(CNC(C2CC2[N+](=O)[O-])=O)c1 C(=O)(C(C)Cc1ccc(CC)o1)NC1CN(C(CCOCC#C)=O)C1 N1(C(C2CC(SC)C2)=O)C2CCCC1CC(NC(=O)C(C(C)C)C(C)C)C2 c1(C(=O)NCCC2CC(NC(=O)CC=C(Cl)Cl)C2)cccc(C#CCO)c1 C1(C(=O)NCC2CCN(C(C3(CSC)CC3)=O)C2)CC12C1CC3CC(C1)CC2C3 c1(CC(=O)N(CC(=O)NC2COC(C(F)F)C2)C2CC2)cnn(CO)c1 N1(C(C(COC)OC)=O)CC2CC(NC(C3(C)CC=CC3)=O)CC2C1 Cc1cc2c(cc1C)OC(C(=O)NCCCNC(=O)Cc1cccc(O)c1)C2 c1(N(C)C)nc2ccc(C(=O)NCC3CC(N)CCO3)cc2o1 N12CCC3(CC3C(=O)Nc3nocc3C1=O)C2.CC(C)(C)SCC(N)=O CC1=C(C(=O)N2CC(CO)(NC(c3snnc3C(C)C)=O)C2)C(=O)OC1(C)C c1(N2CC(OC)C2)ncnc2[nH]cc(I)c12.c1(C=O)cccc(S(C)=O)c1 CC1=CCC(C(N2CC3CC3C2CNC(=O)Cc2cnc[nH]2)=O)CC1 Cn1ncc2ncnc(NCC3CCCCN(C(c4c[nH]c(C(N)=O)c4)=O)C3)c12 c1(C(=O)NC2C=CCN(C(CCSCCCC)=O)C2)cnc2cc(C)nn2c1C c1(CNC2(SC(c3nnnn3C)C)CC2)cscn1.C(C)(C)(C)OC(=O)N N1(C(C(CCNC(=O)CCC(C)CN(C)C)OC)=O)CC2CCN(C)C2C1 c1(C(C)NC(C2N(C(C=C(C)C(C)C)=O)CCC2)=O)c(C)noc1C Cc1cc(C(=O)N(C)CC2CCCCN2C(=O)CCCNC(N)=O)nn1C C12(CNC3CCN(C(CCC)=O)CC3)CC(C)(C1)OC2CO CC1(C)C(CC(N2CC3CC2(C(N2CC(C)(O)C2)=O)C3)=O)CC1O C12(CNC(C(C)OCCOC)=O)CC(NC(c3cnsc3)=O)(C1)C2 C(c1ccc(Cl)cc1)=CC(=O)NCC1(F)CC(NC(=O)C=CC(=O)N(C)C)C1 C1(C(C)(C)NC(C(C)OCC=C)=O)CCCCN1C(C1CCC(C(N)=O)CC1)=O N1(C(C(=O)Nc2cccc(-c3nc(C)[nH]n3)c2)=O)CCC(C2(O)CC2)CC1 C(CC(CC)C(=O)NCCCOCCNC(=O)CC1(C)CCOCC1)=CC Cc1cc(Br)c(CS(=O)Cc2nc(-c3ccccc3)no2)s1 C1(C(N(C2CN(C(c3cc(C)sc3)=O)CC2F)C)=O)CC(C)CCC1C(C)C C1(C(N2CC(CNC(C(C)OCCC(C)C)=O)C2)=O)CC2(C1)CS(=O)(=O)C2 N1(C(CCC2CCC(NC(C3(OC)CCC3)=O)C2)=O)CCC12CC(C(N)=O)C2 c1(N(CCNC(=O)C(F)C2CCC2)CC)ncnc(OC)c1OC C1(CC(=O)NCCC(C)N(C)C(=O)NC2CN(C3CCOCC3)C2)OCC1(C)C c1(C(=O)NCC(CNC(c2c(C)cc(=N)[nH]c2)=O)O)ccnc2ccc(F)nc12 Cc1ccc(Cl)cc1OCCCC(=O)N1CC(CCNC(=O)C2=NOC(C)C2)C1 c1(N2CCCC(CC=C)C2)cc[nH]c(=NCCC(C)CCCO)n1 c1(CC)cc(F)ccc1CC(=O)NCC1CCC1NC(=O)C=C(C)c1ccsc1 c1(C(=O)NCC23C(CN(C(CNC(=O)NC)=O)C2)C3)cc(C)nc2ccnn12 c1(C(N2CCCC(NC(c3c(=N)cc[nH]c3)=O)C2)=O)cnn2c1OCC(F)C2 C1(c2ccc(OC)cc2)CC(C(=O)NCC2(O)CC(NC(=O)C=CSC)C2)=NO1 C(=O)(C1=CCCSC1)NC1(CCNC(C2(C)CS(=O)(=O)C2)=O)CC1 c1(-c2cn(-c3c(C)n(-c4ccccc4Cl)nc3)nn2)cccc2cccnc12 CCC(CN(C)C)C(=O)N1CCC(CC(=O)N(C(C)COC)CCOC)CC1 CC1CC(=O)NCC1C(N1CC(C)(C(=O)NCCSC(C)(C)C)C1)=O N1(C(C(C)(C)C)=O)CCN(C(C2CCN(C(=O)CN3CCNC(=O)C3)C2)=O)CC1 c1(C(N2CC(NC(c3n(CC=C)ccc3)=O)C(O)C2)=O)ncc(N)cc1C c1(-c2cc(C)c(Br)cn2)nc(C2CCCO2)nn1C1CCc2ccccc21 Cc1cc(C#N)cnc1C(=O)NC12CCN(C(c3ccc(CO)o3)=O)CC1C2 C(=O)(C(CC(C)C)NC(=O)CCC1(NC(=O)CC2CCCO2)CCC1)OCC c1(C(=O)Nc2nc3ccc(F)cc3s2)c[nH]c2cc(C(F)(F)F)ccc2c1=O C(N=c1[nH]c(=NCCC2CC=CCC2)[nH]c2c1CCC2)c1cn(C(C)(C)C)nn1 N1(C(CCC)=O)CC(CNC(C2(c3ccccc3)CCOC2)=O)C(C)C1 C(=O)(CCCCC(=O)NC1C=CC(CNC(=O)Cc2c(C)nn(C)c2C)C1)OC c1(OC)cc(F)c(C(=O)NCCC(C)NC(c2ccnc(CO)c2)=O)c(F)c1F C#CCC(C(=O)NCC(=O)OC)NC(c1csnn1)=O N1(C(CN(C(=O)OC(C)(C)C)C2CC2)=O)CCN(C(c2cccc(N)c2)=O)C2CC12 N1(C(c2c(CC)nn(C)c2Cl)=O)CCCC2(CCC(NC(=O)C=C(C)Cl)C2)C1 CC1c2ccccc2CC1C(=O)NC1(C)CN(C(=O)C2=CCCOCC2)C1 C1(C(N2CC(OC)C(NC(=O)C3=C(C)OCCS3)C2)=O)CCn2c(C)cnc2C1 c1(C(N2CCCC2c2ccsc2)C(=O)NC2(C)CC2)cnc(C2CC2)o1 C(N=c1[nH]c2c(c(=NC3CSc4ccccc43)[nH]1)COC2)c1c(C)occ1 c1(C(=O)NC2C(NC(c3cc(C)on3)=O)CCC2)cc(C(C)(F)F)ccc1C C(=O)(C1=CC2C=CC1C2)NC1CCC(CCNC(c2c(C)nncc2)=O)C1 C=C(C)CCCC(=O)NCC1CCCCCN1C(=O)C(CC)n1ccnc1 C1(NC(C(C=C)(C)C)=O)CN(C(=O)CCN(C)CCO)CC12CC2 N1(C(=O)CCc2nc[nH]n2)CCC2(CCCN2C(c2cc(=O)cc(Cl)[nH]2)=O)C1 C(CC(CC)C(=O)NCC1CCN1C(=O)COCc1cc(C)no1)=CC N1(C(C(C)=C2CC2)=O)CCOCC(NC(c2cnnn2C2CC2)=O)C1 CC1(NC(C2CN(C3C(C)C3)C(=O)C2)=O)CCCN(C(C2CCC(F)CC2)=O)C1 C1(NC(C=CCC(C)(C)NC(=O)C=Cc2ccncc2)=O)CCC2CC1CO2 N1(C(=O)CC2CC=CC2)CC(NC(=O)CCOCc2ccccc2)C(O)C1 C1(CC(=O)NCCCNC(C(C)C)=O)C2CCCC2N1C(C1CCOC1C)=O N1(C(CC(CC)OC)=O)C2CCC1CC(C(=O)NC(C)C(F)(F)F)C2 C12(NC(CS(=O)(=O)NC)=O)CCOCC1CN(C(c1ccc(C#N)cn1)=O)C2 Cc1cc(C(=O)NC2CCN(C(=O)C#CC3CCC3)CC2CO)n2nccc2n1 n1(CC)cnnc1CCNC(=O)C(F)CC1CN(C(C2(C(C)(C)OC)CC2)=O)C1 c1(C(=O)NC(C2CN(C(COc3cn(CC)nc3)=O)C2)C)cccc(OC)c1 c1(CC)cc(C(=O)N(C(C)C(=O)NC2CC(n3cccn3)C2)CC)n[nH]1 C1(CNC(C(=Cc2ccncc2)C)=O)CC2COCC2N1C(C1CC(C)(F)C1)=O C(=O)(C(C#N)C(C)(C)C)N(CCNC(CCC(C)OC)=O)C C1(N2CC(CC(C(=O)N(C(C)CCn3cncn3)C(=O)C(Cl)Cl)F)C2)CCOCC1 C=C(C)C1OCCCC1C(=O)NC12CCCN(C(=O)C(C)(C)C#N)CC1C2 c1(C(N2C(CNC(CC(CC)OC)=O)CCCC2)=O)c(N)sc(C)c1C CC(C)C(C(C)NC(C1CN(C)C1)=O)NC(=O)CCn1cccnc1=O c1(C(N2CC(NC(C(c3c(C)cccn3)(F)F)=O)C2)=O)cc2c(nn1)CCCO2 CCC(CN(C)C)CC(=O)NCC1(F)CCN(C(c2ocnc2C(F)F)=O)CC1 C(C1CN2CC1C2=O)=CC(=O)NC1CCCC1.C(C(C)N(C)C(C)=O)SC c1(-c2nnc(N(C)NCC)n2CCOC)ccc(OC)c(OC)c1 CN(C)S(=O)(=O)N1CCN(C(C2CCC3(CCC3)O2)C(=O)NCC2(C)CC2)CC1 c1(C(C)C)ccc(O)c(C(N2CC3CC3(NC(c3cccn(C)c3=O)=O)C2)=O)c1 c1(C(=O)NCC2CN(C(=O)Cn3cnc(Br)c3)C2)ccc(OCCF)cn1 N1(C(C(CNC(c2c(C)cccc2F)=O)C(C)C)=O)CCN2CCC1CC2 CC(N=c1nc2c(cnn2C)c(NCC2(CC#N)CC2)[nH]1)c1ccc(Cl)cc1F C#CCC(C(=O)N1CC(c2cc(O)no2)C1)NC(c1sccc1Cl)=O S(=O)(=O)(c1cc(C#N)ccc1C)N1C(CN2CCC(C(=O)OC)C2)CCC(C)C1 c1(C(N2CC(C)(NC(c3cc(C(C)=O)on3)=O)C2)=O)ccc(CC2CCC2)cc1 CC1(C)CC(NC(c2cnsn2)=O)CN1C(C1CCN(C2CC2)CC1)=O CCCCC(O)CC(=O)NCCCN(C(=O)CC1COCCN1CC)CC c1(CNC(C2(C)N(C(Cc3onc(C)n3)=O)CC2)=O)ccc(Br)cc1 C(=O)(CCCCCCCCCCCC)NCCC(=C)CNC(=O)CCC(C)(F)F CC(C(=O)NC(C1(O)CN(C(=O)CCC(=O)c2cccc(F)c2)C1)C)C(F)F C1(CNC(C(c2cccc(Cl)c2)C)=O)CCCCC1NC(=O)Cn1nnc(=O)[nH]1 C(=O)(CC1=CCOCC1)NCC(C(C)C)NC(c1ncoc1-c1ccco1)=O N1(C(C(CO)N(C)C)=O)CCC(O)(CNC(c2snc(O)c2Cl)=O)CC1 c1(C(N2CC(CNC(c3ccncn3)=O)CC(C)C2)=O)cnc2[nH]nnc2c1 c1(C(=O)NC(C=C)CO)ccc2[nH]c(NC(=O)Nc3ccc(Cl)c(I)c3)cc2c1 N1(c2cc(N(C)C)ncn2)CCN(C(c2cc(I)ccc2O)=O)C2CC12 c1(Cn2cc(C3N(C(CC(=O)OC(C)(C)C)=O)CC3)nn2)ccnc2[nH]ccc12 C=CCCCCCC(=O)NC1CC(C)(NC(=O)Cc2csc(C(C)(C)C)n2)C1 N1(C(C2N(C)CC2)=O)CC2CC(O)C1C2NC(=O)C=C(Br)Br N1(C(c2csnn2)=O)CCCC1CCc1cn(C2CC2)nn1 C(CN=c1[nH]cnc(Cl)c1C#N)(C1CCCC1)NC(c1n(CC(C)C)ncc1)=O C(=O)(NNC(=O)C(C)(C)c1ccccc1)c1c(CN(CC)CC)cccc1 C1(NC(c2cc(OC)ns2)=O)CCCN(C(=O)Cc2ccoc2)CC1 c1(C(N(C)CCNC(C2CCC23CCC3)=O)=O)cc2c([nH]1)CCCC2 c1(C(C)NC(C(CC)SC)=O)ccc(CNC(=O)CCc2ncc(C)[nH]2)cc1 S(=O)(=O)(c1cccs1)NC(C(=O)NCC(CO)NC(CC(C)CF)=O)C C(=O)(C(F)CCC(C)(C)C)N1CC2(C(NC(C(CCC)F)=O)CCC2)C1 C(=O)(C(C)(C)CCCNC(c1ccc(C(N)=O)[nH]1)=O)NCCc1cnc(C)[nH]1 C1(C(=O)Nc2ccc(CCC)cc2)CC12CCN(S(=O)(=O)CC1CC1)C2 N1(C(CN2CC(CC)OCC2)=O)CCS(=O)CC1c1ccc(C)o1 Cc1cc(CNC(=O)NCCN2CCN(Cc3ccccc3)CC2)c(Br)o1 C1(C(=O)NC23CC(CNC(C4N(C)CC4)=O)(C2)C3)CCCC1C1CC1 Cc1c(C(N2CCCC(c3ccncc3)CC2)=O)cc([N+](=O)[O-])cc1[N+](=O)[O-] N1(C(c2c(C)cns2)=O)CCC(C(=O)NCCCF)(CF)C1 N#Cc1cc(CN2CCC(C(F)(F)F)CC2)cc(C(F)(F)F)c1 CCCC(C)(O)CC(=O)NC1(CCCNC(C2(O)CCC(C)(C)CC2)=O)CC1 C(=O)(CCCCCCCC1CC1)N1CCC(N(C(CN(C2CC2)CC)=O)C)CC1 c1(C(N2C(C)CCC(NC(c3cnc(CC)s3)=O)C2)=O)cnc2[nH]c(O)nc2c1 C1(OC)CC2(C1)CN(C(=O)C(CC(N)=O)NC(c1csc(F)c1)=O)C2 C1(NC(C(C=CCCC)O)=O)CCN(C(c2cnc(C(F)F)c(C)c2)=O)CC1C CCCC(CCC)C(C)(c1nnnn1CCC1CC1)NC1CC2CC2C1 c1(CNCc2n(COC)ncc2)ccc(OC)c(OC(F)(F)C(F)F)c1 c1(NC(N(C(CC(CC)C)C)C)=O)c2c(nn1C)CN(C(=O)OC(C)(C)C)C2 C12(NC(c3c[nH]cc(F)c3=O)=O)CN(C(c3cc[nH]n3)=O)CC1CS(=O)(=O)C2 C(C1=CCN(C)CC1)NC(CCCC1CCCN(C(CCSCC)=O)C1)=O C(CC(F)(F)C(F)(F)F)(C(=O)N=c1nc(-c2ccccc2Cl)o[nH]1)OC c1(C(=O)NC2C(NC(C(c3cscn3)N(C)C)=O)C2)cccc2c1OCC2 C=C(C)CCCC(=O)N1CCN(C(c2cc(CC)cc(F)c2)=O)CC1C CC1CCc2n[nH]cc2C1C(=O)NCC1CC(NC(c2ccc[n+]([O-])c2)=O)C1 c1(C(=O)NC(C(=O)N2CC(C(=O)NCC)C2)C(C)OC)ccc2cc[nH]c2c1 C1(COC)CCn2ccnc2C1.C1(C)(C)CC(=O)N1 N1(C(C2CN(C(N)=O)C2)=O)CC(O)CCC1C(N1CC(O)C(O)C1CO)=O c1(NC(C(c2cc(C)cc(Br)c2)N2CCC(O)C2C)=O)ccc2c(c1)OCO2 C1(F)(CNC(CC2CN(C)C2)=O)CCC(NC(=O)CCSCc2ccccn2)C1 Cc1ccc(C(=O)NC(C)(CNC(=O)C(O)Cc2ccc(Cl)cc2)CO)cc1C N1(C(c2c(OC)nc(C)cc2)=O)CCC2CCN(C(C3CN(C)C3)=O)C2C1 Cc1ccc(SCCC(=O)N(CC(=O)OC(=O)CCc2cnc(O)[nH]2)C2CC2)cc1 C(C(=O)NCC(CCNC(=O)CNC(c1ccccc1)=O)OC)(C(C)C)SC N#Cc1c[nH]c2ccc(C(N3CCC(F)(CNC(C4CC4(F)F)=O)C3)=O)cc12 CCC(F)(C(=O)OC)C(=O)NCC(C)CNC(C1(Sc2ccccc2)CC1)=O c1(C(=O)NC2C(CNC(COCCOCC)=O)CC2)nccc2nn[nH]c12 C1(CNC(CC(=C)C)=O)CC2CCC1N(C(C1CC=C(C)CC1)=O)C2 N1(C(C(CC)C(=O)OC)=O)CCOC2CN(C(c3cc(C(C)(C)C)[nH]c3C)=O)CC12 c1(SC(C(N2CC(NC(C(CCCC)O)=O)(CO)C2)=O)C)nc2ccccc2s1 S(=O)(=O)(c1nc(N2CC3CCC(C2)C3O)ccc1Br)N(C)C c1(C(N2CCCC(CN(C(C3(CC)CC3)=O)C)C2)=O)cnc2c(c1)NC(=O)CS2 C(=O)(CS(=O)(=O)CCO)N(CC(C)NC(=O)CC1CC(C)=NO1)CC C12(NC(CCCC#C)=O)CN(C(=O)CCN3CCCCC3=O)CC1CS(=O)(=O)C2 c1(CN(C(=O)CC2CCC2)CCNC(C2CC23CCC3)=O)ccccc1 N1(C(=O)Nc2cccc(N3CCOCC3)c2)CC2CN(c3ccncn3)C2C1 C(C(C)(O)CC(=O)N1CC(n2cc(-c3ccc(N)cc3)nn2)C(C)C1)OC c1(CC(=O)NC23CC(CNC(=O)CC4CCCCC4)(C2)C3)ccc2occc2c1 C1(N(C)C(c2csc(CNC(C3CSCCS3)=O)n2)=O)CCCCCC1 c1(OC)cc(C(N2CC(OC)C(NC(C3CC(OC)C3)=O)C2)=O)cc(N)c1O C(CC(C)CCNC(=O)Cc1ncc(C)s1)NC(c1c(CC)noc1)=O c1(CCNC(C(=O)Nc2nccc(OCCOCC)c2)=O)nnc2n1CCC2 c1(C(=O)NCC2N(Cc3c(C)scn3)CCC2)nc2ccc(F)cn2n1 c1(OC)nc(N2CC3CC(NC(C4COC(C)C4)=O)CC2C3)nc(C)c1F c1(C(N(C(CNC(C(C(CC)C)C)=O)C2CC2)C)=O)cccc2c1CCCC2 N1(C(C(C)(C)C(F)(F)F)=O)CCOC2(CCN(C(=O)C=C3CC3)C2)C1 C1(CC(=O)N(CCN(C(=O)C(=O)N(C)C)C(C)C)C)CCC(=O)N1C c1(C(N2CC(NC(CN3CC(C)C3)=O)CC3(C2)CC3)=O)nnc2ccccc2n1 C(=O)(C(C)CS(C)=O)NCC#CCNC(c1cc(CC)no1)=O c1(SCCOc2n(C3CC(C(=O)OC)C3)c(C)c(Cl)n2)ccc(Br)c([N+](=O)[O-])c1 Cc1nn(C)cc1C(O)C(=O)NCC1C2CN(C(C3(NC(N)=O)CC3)=O)CC12 C1(C(=O)NC(CC)(C)CNC(=O)CCc2cscn2)CC12CCCC2 C(CC(C(=O)NCC(C)CC1CCC1)NC(=O)CC1CC(OC)C1)=CC c1(C(N(CC(CC)NC(C2(OC)CCC23CCC3)=O)C)=O)cnn2ccncc12 N1(C2CCN(C(C)C)C2=O)CCC(NC(C2CC23CCOC3)=O)CC(C)(C)C1 N1(C(=O)NC2(CC)CC(O)C23CCC3)CC2(CCCCC2)C1C(C)C N1(C(Cn2c(C)ccn2)=O)CCC(C(=O)NC(C)Cc2nncn2C)C1C CC(C)C(F)C(=O)NC1(CNC(=O)C(c2ccc(F)cc2)=O)CCOC1 Cc1cccc(C(=O)NC(C2(O)CN(C(=O)C(O)CN3CCOCC3)C2)C)c1F c1(C(N(CC(C)(C)NC(=O)Cn2nc(O)ccc2=O)C)=O)cc2n(c1)CCOC2 c1(C(=O)NC(CN(C)C(c2n[nH]cc2Cl)=O)(C)C)cc(OC(F)F)cc(Cl)c1 N1(C(c2cc(C)nc(Cl)c2)=O)CCOC2(CCN(C(=O)C(F)(F)C(F)F)CC2)C1 CCC(CC(C)C)C(=O)NC1(C2CN(C(c3cncc(C)c3)=O)C2)CC1 N1(C(C2(C#N)CC(C)C2)=O)CC2CCCC2(NC(c2cnc(C(F)(F)F)s2)=O)C1 c1(C(=O)NC(C2CCN(Cc3cc[nH]c3)CC2)C)ccc2nc(Br)sc2c1 C#Cc1ccc(Br)c(C(=O)NCC2CC(NC(=O)C(C)c3ccsc3)C2)c1 c1(N(CCCN(CC(N)=O)C)CC)cc(NC2CC2(C)C)nc(C)n1 C(=O)(CC1=CCOCC1)NC(C(C)NC(CCc1cccc(C(=O)NC)c1)=O)C CC(C)(F)CCC(=O)N1CC(C(=O)N(C2CCC3(CC2)CC3)C)CC12CCC2 c1(OCC)cnc(C(N2CCC(CF)(NC(=O)CC(C)C3CC3)C2)=O)cn1 c1(C2(C(=O)NC(C(=O)OC)CSC)CC2)ccccc1Cl.N1CCCCC1 c1(SC)cccc(C(=O)NCCCOC2CCN(C(c3cc(Cl)ns3)=O)CC2)c1 CCC(CCOC)C(=O)NC1CCCCCC1C(=O)NC(CN1CCCC1)CO c1(C(=O)NCCCCCNC(Cn2c(CCC)ncc2)=O)ncc(Cl)cc1Cl C(=O)(CCCC(F)(F)CO)NC(C)C(CO)NC(C1CCS(=O)(=O)CC1)=O C(=O)(CC1=CCOCC1)c1cn(C2C(C)(O)CCC2)nn1.C12CCCCC1NC2 c1(C(=O)OC(C2CCOCC2)C(=O)OC)ccccc1S(=O)(=O)CCS(C)(=O)=O C1(C(N(C2CCNC2)CCC#N)=O)CC2CNCC(C1)C2=O C(CC(=O)NC(CNC(c1cc(C(C)C)no1)=O)C(C)C)(OCC)OCC C(=O)(C1=CCC(NC(C2C=CCCC2)=O)C1)NCc1n(CCC)cnc1 c1(C(=O)NC2(CC=C)CN(C(c3nonc3N)=O)C2)cc2occc2s1 CCC(CC(=O)NC(CNC(C1CCN(C)C1=O)=O)C(C)C)c1ccc(C)cc1 C1(C(=O)NC(C(=O)OCC)C2CC2)CCC2(CC2)N1C(c1cc(CCO)on1)=O CCCN=C(NCCOc1cccc(SC(F)(F)F)c1)NCC(C)(C)CN(C)C c1(CN(C(=O)NC2CC(C)(C)C2)CC)cncn1C c1(C(C(=O)NC2C(C)CCN(C(=O)C(C)(C)N(C)C)C2)O)cc(F)c(F)c(F)c1 CC1CC(C(=O)NC(C2(O)CCN(C(=O)CNC(=O)NC3CC3)C2)C)CCO1 C1(NC(=O)C2=CCSC2)CC2CCC1N(C(=O)Cn1ccc3ccccc13)C2 c1(C(=O)NC(CCC(=O)OCC)C)sc2ccccc2c1Cc1nn[nH]n1 C1(C(=O)NC(C2CCCN(c3ccnc(C(C)C)n3)C2)C)CC(=O)CC12CCC2 n1(CC(=O)NC(CCN(C(C(CC)CN(C)C)=O)C)C(C)C)nc(O)ccc1=O N1(C(c2c(CC)cccn2)=O)CC(CNC(=O)CCC(=O)NC)C2(CC2)C1 C12(NC(CCC(=O)NC)=O)CCC1CN(C(=O)C(C)CO)C2 c1(CC(=O)NC2(COC)CN(C(CC3(OC)CC3)=O)C2)cccc2ccccc12 c1(CN2CC3C(NC(c4ncc(C)nc4)=O)C3C2)cc(Cl)c(O)c(Br)c1 C1(C)(c2cn(CCC(=O)OC)nn2)CN(C(C2COCCC2(F)F)=O)CCO1 C1(C(N(C2CCN(C(c3c(CC)noc3)=O)C2)C)=O)CC2(CCCCC2)CO1 C(=O)(C(=O)CC(C)C)NC(CCNC(CCC(=O)NCC)=O)C(C)C C(=O)(CC(CC)C(F)F)N1CC(C(=O)NCC=CC)C(CCC)C1 Cc1cncc(-c2cn(CCc3ccc(N(C(=O)C(C)C)C(C)C)cc3)nn2)c1 C12(NC(C3C=CCCC3)=O)CC3CCC(C1C2)N3C(c1coc(O)n1)=O N1(C(c2c(N)sc(C)c2C)=O)CCCCC(NC(=O)CN2CCC(C)(O)C2)CC1 O=C(CC1NCC2CCCC12)N1Cc2ccccc2CO1 C(CN=c1[nH]c(N(C)CCOC(C)(C)C)nc(=N)[nH]1)N1CC(C)CC(C)C1 C1(C(=O)NCCCSCC)C2CCC(C2)N1C(c1c[nH]c(=N)c(C)c1)=O C1(NC(C(COC)NC(C(CC)N(CC)CC)=O)=O)CCCC1N=[N+]=[N-] N1(C(C2C(C)(C)C2(C)C)=O)CC2CCC(CNC(=O)CC(F)(F)Cl)C2C1 N1(C(C(CC(C)C)NC(C)=O)=O)CCC2(C1)CN(C(=O)CCC(=O)OC(C)(C)C)C2 C(=O)(CCC(O)C(C)(C)C)N1C2CC(N(C(C3N(C)CCCC3)=O)C)CC1CC2 N1(C(c2nc(C)c(C)[nH]2)=O)CCCC(CCNC(c2ccncc2F)=O)CC1 C12(C(=O)OC)CCC(C(=O)NC(CC)C(=O)Nc3ccc(Cl)cc3)(CC1)C2 N1(C(C(C2CC(F)(F)C2)OC)=O)CCC(CN(C(=O)CC2CC=CC2)C)C1 c1(C(N2CC=CC2Cn2cc(C3(CO)CC3)nn2)=O)ccc(F)c(Br)c1 c1(NC(c2c(-c3c(NS(C)(=O)=O)cccc3)ncs2)=O)cncc(Cl)c1Cl Cc1cc(C(N2CCC(C)C(NC(=O)COc3ccon3)C2)=O)c(C)nc1C Cc1ccc(CNC(C2CC23CC(NC(=O)Cc2csc(C)n2)C3)=O)cc1 C12(C(=O)NC3CCC(CNC(COCP(C)(C)=O)=O)C3)CCC(CC1)O2 C1(CNC(C(C=C)(C)O)=O)N(C(=O)Cc2ncc(CC)[nH]2)CCCC1(C)C N1(C(C2(CS(N)(=O)=O)COC2)C)CC2CN(c3nccc(C(F)(F)F)n3)CC2C1 N1(CC2CCC(Cl)CC2)CCN(C(=O)NC(c2onc(C(C)C)n2)C)CC1 C1(C(N2CC(CCCCNC(Cc3ccc(C)s3)=O)C2)=O)CCOC(=O)CC1 c1(C(=O)NCC(N(C(CNC(CCC)=O)=O)C)C2CC2)cc(F)c(F)c(C#N)c1 c1(CNC(c2nc(C(C)OC)oc2)=O)ccc(NC(COC)C(=O)C(C)=O)cc1.OC N(C(=NCCCCNC(=O)OC(C)(C)C)NCC1(C(F)(F)F)CCCC1)C(C)C c1(CC(=O)NCC2C(CNC(COCC)=O)C2)cccc(O)c1F N1(C(c2nc(C)[nH]n2)=O)CCC2(CNC(c3ccnc(O)c3)=O)CCCC12 C(=O)(C(CO)C(C)(C)C)N(C(CC(=O)OC)C)Cc1ccccc1 n1(CC)nc(C)c(C(=O)NC2CN(C(c3cncnc3C)=O)C3CC23)c1C C1(NC(COC(C)C)=O)CN(C(=O)CN2CC=CC2)CC1C c1(OC)ccc(CC(C)CNC(c2ccccc2-c2cncnc2)=O)cc1 c1(CC)cc(C(N2CCC(CN(C)C(C34CC(C3)C(C)(C)O4)=O)C2)=O)c(C)nn1 c1(CN(C(C23CCCC(CC2)N3)=O)CC)cc2ccccc2o1 Cc1cc2ccc(C(N3CCC(O)(C(C)CNC(=O)CCC(N)=O)C3)=O)cn2c1 C1(C)(NC(C(N2CC(C)C2)C)=O)CCCC1NC(c1ccc(CCO)cc1)=O CC(CN(C)C)CC(=O)NCCC1(O)CCN(C(=O)Cc2ccn(C)n2)C1 c1(C(=O)NCCC2CCN(C(C3COCCO3)=O)C2)cccc2c1CCCCC2 N1(C(=O)Cc2cc(C(F)(F)F)ccc2Cl)CCSc2c([nH]c3ccccc23)C1 Cc1scnc1C(=O)NC(C)C(C)NC(=O)C=CCN1CCCC1 C(C1C(C(N2CCC(CC(N)=O)CC2)=O)C1(C)C)=C(C)C.N12CCCC1CC2 N1(C(CCC#C)=O)CCCC12CCCN(C(C1(CCO)CC1)=O)C2 C1(NC(C(C)NC(=O)C(F)(F)C2CCCC2)=O)CCN2CCCC12 C(=O)(CC(C)C(F)F)N(C1CCCN(C(C2C(C(C)=O)C2(C)C)=O)C1)CC1CC1 c1(C(=O)NCC(C)CNC(C2CCCC2C(F)F)=O)ccc2c(c1)NC(=O)CC2 c1(NCC(C)(C)C(F)(F)F)nc2ccccc2nc1NCc1ccc(F)cc1Cl Cc1ccc2c(c1)NCCN(C(=O)C1=CC3CCC=CCCC13)C2 C(=O)(CN=c1[nH]c(N2CCC(CN(C)C)C2)nc(=NC)[nH]1)NCCC C1(NC(=O)CC=C(Cl)Cl)CN(C(c2cnn(C(F)F)c2)=O)CCC1O c1(OC)ccccc1-c1oncc1C(=O)N(CC(C)N(C(=O)C(C)C1CC1)C)C CC1CCN(CC(=O)NCC(C)(C2CCC2)NC(=O)Cc2ncc(Cl)s2)C1 c1(C(N2C(C(=O)OC)CCC2C(C)C)C(=O)NCCSC)ccc(C#N)nc1 N1(C(c2c(C)oc(-c3ccccc3)c2)=O)CCCC(C)(NC(=O)CSC(C)C)C1 N1(C(C=C(C)c2ccsc2)=O)CC2(CCCCN2C(=O)CC2CCOC2)C1 c1(OCC(N2CC(C(C)NC(C3CC34CC(C)(C)C4)=O)C2)=O)cccc(F)c1F C(CC(C)C)(C(=O)NCC1(NC(c2ccc(C)s2)=O)CCCCC1C)OC C#CCC(O)C(=O)N1CC=CC1(C)C(N1CC(OCCO)C1)=O Cc1nn[nH]c1C(=O)NC(C)(C)CN(C)C(C1CCCC1O)=O c1(C(N2C3C(CNC(CCC(C)SC)=O)C(C3)C2)=O)coc2ccc(Cl)cc12 C1(NC(CNC(=O)CC(F)(F)F)=O)CN(C(=O)C(F)n2cccn2)C2(CCC2)C1 O(NC(=O)C(CNC(=O)Cn1ncnn1)C(C)(C)C)CCCCC C1(CNC(=NCC2C(C(=C)C)OCC2)NCC(C)(C)OC)OC(=O)CC12CCC2 C(C1CC1)(C1CC1)=CC(=O)NC(C(N1C(CCN(C)C)CCC1)=O)C1(O)CCC1 C(CC(=O)NC(c1snnc1C)C)(C(F)(F)F)NC(c1ccn(CCC)n1)=O c1(N(CC(C)CNC(C2CCOC(C)C2)=O)C)ncc(C#N)cc1F C1(O)(CNC(c2cc(F)cs2)=O)CCCN(C(=O)C=Cc2cnc[nH]2)CC1 N1(C(c2n(C)nnc2)=O)CCC(C(N2CCOC3CC23)=O)CC1(C)C N1(c2ncc(-c3ccc(C)cc3)cn2)CCC(F)C(NC(C2CC2(C)C)=O)C1 Cc1nc(-n2nc(COc3cccc(Cl)c3)nc2C2CCC2C)n(C)n1 CON1CCC(C(=O)NCCCN(C)C(C2CCC(C3CC3)C2)=O)CC1 S(=O)(=O)(c1ccccc1Br)N1C2CN(C(Cc3ccc(OC)cc3Br)=O)C(C2)C1 N1(C(C2C(NC(c3cc(I)c(O)c(I)c3)=O)C2)=O)CCC2(CCCOC2)C1 C1(CNC(C2(COCC)CC2)=O)CC2CC(C1)N(C(=O)C#CC(C)(C)C)C2 c1(CC)ccc(C(N2CCC(O)C(NC(c3cc(Cl)ns3)=O)C2)=O)cc1N C1(C(N2CCC(C(C)NC(C3CCCNS3(=O)=O)=O)C2)=O)CC2(COC(=O)N2)C1 C1(C(=O)NC2C3CCN(C(c4ccc(C)c(C)n4)=O)C32)CCCC(F)(F)CC1 c1(C(N2C3CCC2CN(C(C2CC2C2CC2)=O)C3)=O)ccc(F)c(F)c1Br C1(C(N2CCCC(C(=O)NCCc3cn[nH]c3)C2)=O)OCC2CCCC12 C(=O)(CC(C(C)C)NC(=O)CCC1CCCC1)NCCn1c(C)nnc1 CN1CCN(C(C2CCC3(CC2)CC3)=O)CC1CNC(=O)CCF c1(CC)cccc(C(N2CCCC2CN=[N+]=[N-])C(=O)NCCC#N)n1 N1(Cc2c(-c3ccc(C=O)cc3)cccn2)CCC2(CCCO2)CC1 N1(C(C(C)C2CCCC2)=O)CC(N(C(=O)Cn2ncnn2)C)C2(CC2)C1 C1(C(=O)NCC2C(NC(CNC(=O)C3CC3)=O)C2)CC2(C1)CC2F CC(C)CC(O)CC(=O)NCCC(F)Cn1cc(-c2cc(Cl)cc(Cl)c2)nn1 c1(N2CCC(C(C)C)C2)nc(=NCC2(CO)CC3CC3C2)[nH]c2c1COCC2 N1(C(C2(C)CC(C)C2)=O)CCC(OCCCNC(C2CC(C(C)C)C2)=O)CC1 C1(C)(CC)CN(C(c2cc(-c3cccc(F)c3)on2)C(=O)NC(C)(C)C)CCO1 c1(SCC2(C(=O)NC3CCN(C(CC=CC)=O)C3)CCCO2)ccc(F)cc1 c1(C(=O)NC2CC(CCNC(C3(C)CS(=O)(=O)C3)=O)C2)cccc2[nH]c(=N)oc12 c1(OCC)ccc(C(=O)NC2(C)CCCN(C(=O)C(C)C3CCC3)C2)c(F)c1F c1(N2CCC(NC(=O)NCC3C(C)(OC)C3)CC2)nc2ccccc2o1 c1(C(N2C(CN(C(=O)Cc3nccs3)C)COCC2)=O)nn(C)c(Cl)c1Cl n1(CC(=O)NCC(CO)NC(c2occ(C)c2)=O)nnc2ccccc2c1=O C1(C(C(=O)N(CCCCC)C(C)C)C)CCCN(C(c2ccn(CC)n2)=O)C1 C1(NC(C(CO)OC)=O)CCOC(C(=O)NC(CO)C(F)(F)F)C1 C(CC(=O)NCc1cn(C)cn1)(C1CC1)NC(CC=C)=O c1(C(C(CO)NC(C(c2ccc(F)cc2)C)=O)O)ccc(Br)cc1 N1(C(c2c(C)ncs2)=O)CC2CCC(NC(c3cc(CC4CC4)on3)=O)CC2C1 N1(C(c2c(CC)csc2)=O)CCN(CC(C)(C)NC(=O)C(C)CC2CCC2)CC1 CC1(C)CC(NC(C2(C)CC2(Cl)Cl)=O)CCN(C(c2nc(Cl)cs2)=O)C1 C1(C(=O)Nc2ccc(C)nc2)CN(C)CCN1C(=O)C=Cc1cscn1 C1(C(=O)NCC(CC)(C)NC(=O)Cn2nccc2C)CCN(C(C)C)CC1 C12(NC(COC(CC)(C)C)=O)CCN(C(=O)CCOC3CCCC3)CCC1C2 c1(C(=O)NC(CC)CNC(C2(CC(C)C)CCC2)=O)oc(SC)cc1C Cc1nn(C)c(C)c1C(=O)NCC1CCN(C(c2ccc(F)c(Cl)c2)=O)CC1C N1(C(C2(C(C)C)CC2)=O)CCC2(CC1)C(N(C)C(c1nccn1C)=O)CS2(=O)=O N1(C(C2(OC)CC2)=O)CCCC(NC(c2c(C)nsc2N)=O)C1 CCCCC(C(=O)N(C1CCCCC1)CCNC(=O)CCN(C)C)C(C)C C1(C(N2CCC(C(CNC(C3CCCCC3F)=O)O)CC2)=O)CCC(F)(F)CC1 CCC(CC)CC(=O)N1CC2(CNC(=O)C3=NOCC3)CC1(COC)C2 c1(C(N(CC(CC)NC(C2(C#N)CCN(C)CC2)=O)C)=O)n[nH]c2c1CCCC2 C(CCCCCNC(C1(CNC(=O)CC#N)CC12CCC2)=O)N(C)C C#Cc1ccc(C(C(=O)Nc2ccccc2F)N(C)Cc2cn[nH]c2)cc1 c1(C(N2C(CNC(C(CSC)C)=O)CC(O)C2)=O)ccc(F)c(Cl)c1 CC1(O)CCN(C(=O)CC2(C)CCCN2C(=O)C(F)=C2CCCC2)CC1 c1(C(c2nnnn2C2CC(F)(F)C2)NC(c2nccs2)CC)cnc(O)s1 C1(NC(C=CC=CCC)=O)(CC)CCN(C(C2(C)CCC(C)C2)=O)CC1 c1(-c2nc(C(C)OCC)nn2-c2cc(C)ccn2)ccc(C)cc1CC C1(C(N(CCCNC(C(C(CC)C)OC)=O)C2CC2)=O)CCC2(CC1)CC(=O)C2 CCC(C)(CCNC(=O)CCOCc1ccccc1)NC(=O)C(C)C1CCC1 c1(OCC(N)=O)ccccc1C(=O)NCC(O)CNC(=O)CC1COCCOC1 CC(C)C(CCNC(C1CCNC(=O)C1)=O)NC(c1ccc(Br)cc1)=O C(CCC(O)C(=O)NC1CC(=O)N(CCC)C1)NC(C1(C#C)CCCC1)=O c1(C(N2CC3CN(C(c4c(C)cco4)=O)CC32)=O)c[nH]c2cc(Cl)ccc12 O=C(C1=CCCN(C(C2CCCCC(=O)N2)=O)C1)NC1CCn2ncnc2C1 c1(OC)ccc(C)cc1CC(N1CCN(C(=O)CC2CCSC2)C2CC12)=O CC1CN(C(c2cc(N)c(Cl)c(O)n2)=O)CC(C)N(C(=O)CC2CCC3CC23)C1 N1(C(Cc2nc(C)oc2)=O)CCN(C(=O)C(C(C)(C)C)NC(N)=O)CCC1C C(=O)(C1=NOC(C)C1)NCCNC(C(C(C)O)NC(=O)C1CC1)=O C1(c2cn(C3(C(=O)O)CC3)nn2)(C(=O)NCc2scc(C)n2)CC2(CC2)C1 Cc1ccc(-c2cn(CCC3CC(NC(C4CC(CCO)C4)=O)C3)nn2)cn1 C1(NC(C(CCC)F)=O)CCC2(CCCN(C(=O)COCC(C)(C)C)C2)C1 C1(CNC(c2[nH]cc(C)c2)=O)CN(C(=O)CC2CCC(F)(F)CO2)CCC1(F)F C(CC(C)(C)C)(C(=O)NC1CC(C)(CO)C1)NC(C=Cc1c(C)cccc1)=O N1(CCC(=O)NC(CN2CCC(C)C2)=O)CCN(C)CC1.C12(CC1)CC2 C1(C(=O)NCCNC(C2(CC#C)CCOCC2)=O)CCC(C(C)C)NC1=O CN1CCC(=CC(N2CCC(CCNC(C3C=CCCC3)=O)CC2)=O)CC1 N(C1CCCc2n[nH]cc21)C(C1C(CC)CCN1C(c1cc(COC)[nH]n1)=O)=O CC(C)(C(=O)NNC(=O)C1(S(C)(=O)=O)CC1)Oc1cccc(C#N)c1 CC1CC2CN(C(=O)C(=O)N(CCC(F)(F)F)C3CCCC3)CC12 N1(C(c2cc(F)n[nH]2)=O)CCC2(CC1)CC2NCCNC(C1(C(F)(F)F)CCO1)=O c1(C(=O)NC2C(CNC(CC(C)OC)=O)CCCC2)cc2c(s1)CC(C)(C)C2 N1(C(CC(CC)C(C)C)=O)CCc2cc(CNC(=O)COC(C)CC)ccc2C1 CCCCS(=O)(=O)N1CCC(C(=O)NCC2CCO2)C1 c1(C(=O)NCC2(NC(=O)CC(=O)NC3CC3)CC(OC)C2)cncn(C)c1=O N1(C(COc2cn(C)nc2)=O)C(CC(=O)NCc2ccc(O)nc2)C2CCCC12 C1(C(N(C2CCSCC2)C)=O)CCN(C(=O)c2[nH]ccc2C2CC2)O1 C1(NC(CC2(CC)CCC2)=O)(COC)CN(C(=O)Cc2cn(C)nn2)C1 c1(SC(C)C(=O)N(CC(C)O)CCNC(C2(C(C)(F)F)CC2)=O)ccccn1 C1(COC)(NC(=O)Cn2nnc(C)n2)CCCN(C(C2(O)CCC2)=O)C1 CCC(C)CC(C)C(=O)Nc1ccc(CCn2cc(C3CCCN3C)nn2)cc1 C1(C(N2CC(CNC(C3C(OCC)CCC3)=O)C(C)C2)=O)(OC)CCCCCC1 C1(C(=O)NC2(CC(C)C)CC2)(NC(C2COCCO2)=O)CCC(C)(C)C1 Cc1cccc(C)c1C(=O)N(CC(C)CNC(=O)C(C)(C)c1ccccn1)C CN1CCN(C(C2CC(N(C)C)C2)=O)C(C(=O)NC2CC(C)(O)C2)C1 C1(CC)(NC(=O)CCC2CC(NC(=O)C(C)NC(=O)C3CC3)C2(C)C)CC(C)(C)C1 N#Cc1csc(CC2(C(=O)Nn3cc(C4CC5CCC4C5)nn3)CC(F)(F)C2)c1 C(=O)(CCCCCCCCCO)NCCC(C)NC(C1CCC2(CC2)C1)=O c1(CC(=O)NC2CCN(C(C(CC)(C)OC)=O)C2)ccc(OC(C)=O)c(OC)c1 c1(COC)ccccc1-n1cc(C2(NC(C3CC(F)(F)CS3)=O)CCC2)nn1 C1(N(C(C(=O)NCc2nc(Cl)cs2)C2CC2(C)C)C)CCCCC1 CCCCC(C)C(=O)N1CCC(CO)(CNC(C2(N(C)C)CCC2)=O)C1 C12CCCCCC1NC2=O.c1(C(C(=O)NCC2CC3CC3C2)O)ccc(F)cc1 C(CC(=O)NC(CO)C1CCC1)(C(F)(F)F)NC(CN(C(=O)OC)C)=O C(=O)(C(CC(C)C)N(C)C)N(C(C)CNC(c1cnc(O)n1C)=O)CC N(C1CN(C(c2ccc[nH]2)=O)Cc2ccccc21)C(CC(C)C(C)(C)C)=O CCCCC(C)(F)C(=O)N1CCC(F)(CNC(c2n[nH]cc2C(=O)OC)=O)CC1 C1(C)(COC)CC(NC(C2CC2OC(C)(C)C)=O)CN1C(c1ccn(CF)n1)=O CC(C)S(=O)(=O)CC(=O)NC1CCCCC1CNC(C1CCCC12OCCO2)=O CCCCC(CO)NC(C1CN(C(=O)Cn2cccnc2=O)CC1F)=O CCCCC(=O)C(=O)N(C1C2CN(C(c3cscc3Br)=O)CC12)C Cc1oc2ccccc2c1CC(=O)N(C1CCS(=O)CC1)C N1(C(c2n(CCC)ccc2)=O)CCCC2CN(C)CC12 CCC(C)(C)CN=c1nc2c(ncn2C)c(NC2CCCC3(CC2)CC3)[nH]1 S(=O)(=O)(c1ccc(C#N)c(N2CCC(CCCO)C2)c1)NC1(CCC)CCOC1 c1(CN2C(C(=O)Nc3cc(Cl)ccn3)CC3CC32)cn2ccccc2n1 N1(C(=O)CC2CC23CC3)CC(O)(C2CCCN2C(c2cc(CO)[nH]n2)=O)C1 n1(CC)nc(C(=O)N(C)CC2CCN(C(C3CC4CC3C4)=O)C2)cc1C N1(C(C2(OC)CC2)=O)CC(CO)C2(C1)CN(C(c1nn[nH]c1C(F)(F)F)=O)C2 C1(C(N2CC(CS(C)=O)C2)=O)CCC2CCC1N2C(=O)CS(C)(=O)=O c1(C(N2CCC(CCNC(CS(C)(=O)=O)=O)C2)=O)ccc(Br)cc1N(C)C C1(C(C)(C)O)(CNC(CCNS(C)(=O)=O)=O)CN(C(=O)CCCF)C1 N1(C(C=Cc2cn(C)nn2)=O)CC2CC(NC(c3cc[n+]([O-])cc3)=O)C1C2 Cc1[nH]c(C)c(C(=O)NC(C)CN(C(=O)C(c2ccc(Cl)nc2)(C)C)C)c1C CCC(CNC(=O)C(CC)NC(C)=O)N=c1nc(CC2CC2)[nH]s1 C1(NC(C2C(OC)(OC)CC2)=O)CCC(NC(=O)CSc2nccn2C)CC1 C1(CC(N2CCOCC(NC(c3cocn3)=O)C2)=O)CCc2sccc2C1=O C(C(C)(C)C(C)(C)C)NC(CNC(CNC(C(C)C1CCCC1)=O)=O)=O N1(C(c2cnc(OC)nc2)=O)CCC(CNC(c2cnco2)=O)C(C)C1 C12(C(=O)NCC(CC)NC(=O)C=C(C)C)CCOC1CN(C(=O)NC(C)(C)C)C2 Cc1ccc(O)cc1CNC(=O)COC(C)(C)CNC(C1CC2CCCC2C1)=O N(C(=NCC(c1ccccc1F)N(C)C)NC(C)(C)C)CC(C)C C(CC(CNC(=O)COc1ccccn1)OC(C)=O)OC C1(=O)C2=NN(C(=O)CC2)CC(=O)O1.c1(CC(=O)NCC(C)NC(N)=O)ccsc1 C1(c2nnnn2CC)(NCc2ccc(CC)o2)CC2(CCCCCC2)C1 c1(CC(=O)NC(C)(C)CNC(C2CCC(C(F)(F)F)O2)=O)cc(Cl)nc(Cl)c1 N1(C(C(C)NS(CC)(=O)=O)=O)CC(CNC(C2(C)CC(C)C2)=O)(OC)C1 C(CC(C)C)(C(=O)N1CCN(C(=O)COCC2CCCOC2)C(C)C1)NC(C)=O Cc1cc(C=CC(N2CCC(CN(C(=O)CCc3cnc[nH]3)C)C2)=O)c[nH]c1=N C(=O)(C1=CCCCC1)N1CC(O)(C(C)NC(C2CCC(C)O2)=O)C1 C(N=c1cc(C)[nH]c(=NCC2CCCC2C)[nH]1)c1ncc(CC)o1 Cc1ccc(C(c2nnnn2C2CCCC2)NCc2ccc(Cl)o2)cc1[N+](=O)[O-] N1(C(C=CC)=O)CCN(C(c2ccc(C3CCCCC3)cc2)=O)C2CCCC12 N1(C(c2cc(F)c(Br)cc2F)C(=O)NCCC)Cc2nn(C)c(C(=O)OC)c2C1 c1(NCC(=O)NC2C(NC(CCC=C)=O)CC2)cccc(C#N)c1 N1(C(C(C)NC(C)=O)=O)CC(NC(=O)C(C)(C)n2cncn2)CC12CCCCC2 C1(CNC(Cn2c(CCC)ncc2)=O)CC2CCC1N2C(=O)C(C)(C)N(C)C c1(-c2ccc(C(=O)NC3CCCC3)c(F)c2)cc(F)c(C(N2CC3CCCC2CC3)=O)c(F)c1 Cc1ccccc1C(=O)NCC(=O)NCC12CC1CN(C(C1(O)CCSC1)=O)C2 C1(C(=O)NC23CC(NC(=O)Cc4cccs4)(C2)C3)CCC2(CC1)CNC(=O)C2 c1(NCC(C)C)cccc(C(N2CC3CC3(CNC(C3(O)CC3(C)C)=O)C2)=O)c1 N1(C(c2c(OC)nsc2)=O)CCC(C2CC2)(NC(c2ccc([N+](=O)[O-])[nH]2)=O)C1 N1(C(CCC2C(C)C2)=O)CC(C(N2CC(c3ccccc3)C2)=O)C2(CC2)C1 C12(CNC(C3C(CCC)C3)=O)CN(C(C3CC(=O)NC(C)C3)=O)CC(F)(C1)C2 c1(CC)ccc(C(=O)NC2CC(NC(C3(C)CCC3)=O)C2)cc1[N+](=O)[O-] c1(CC)cncc(C(=O)NCC(O)C(=O)NCC(F)(F)C(F)F)c1 c1(CC)cccc(Cl)c1C(=O)NC1CC1CNC(c1ccc(CC2CC2)o1)=O C(C)(CS(=O)(=O)NC1(CCO)CCOCC1)NC(C(=O)NCC)=O C(=O)(CCS(N)(=O)=O)NCC(CCCC)NC(C1CCC1c1nc[nH]n1)=O N(C1CCc2c(Br)cccc21)C(=O)C(N1Cc2ccc(Br)cc2CC1C(F)F)=O C1(CC)CCN(C(=O)Cn2ncccc2=O)C1CNC(C1CC(F)(F)C1)=O c1(-c2ccc(C(=O)NCCC(C)(C)OC)o2)ccc(C(=O)NC2(CF)CC2)cc1 CCCCC(O)CC(=O)NCC1(CNC(=O)CCNC(=O)COC)CC1(F)F c1(CC2CCCN(C(C(COC)NC(=O)OC(C)(C)C)=O)C2)cccc(Br)c1F C(=O)(CCN1CCCC1)NC.C1CCNC(=O)C2(CC2)CNC(=O)N1CC C1(CC)CC2CCC(C1)N2C(=O)C(O)CCNC(=O)CC(C)(F)F C(CC(C)C)(C(=O)NCCCN(CCCNC(c1ccsc1Br)=O)C)OC CN1CC(O)CC1C(=O)NCC1CN(C(c2csc(-c3ncccn3)n2)=O)C1 CC1=NNC(=O)C1CC(=O)NCC(O)CCNC(C1CCS(=O)CC1)=O c1(C(N(CCOCCNC(CC(C=C)C)=O)C)=O)cn2nc(C)cc2[nH]c1=O c1(C(N(C)CC2CCCN2C(=O)CC2CC2)=O)cc(OC(F)F)ccc1[N+](=O)[O-] C(=O)(C(F)(F)CO)N(C1CN(C(=O)C=C2CCC(C(C)(C)C)CC2)CC1O)C CC(C)(C)C(O)C(=O)NCC1CN(C(c2cccc(C(F)(F)F)c2F)=O)CCO1 c1(C(N2CCC(NC(CCCOCC)=O)C2)=O)cnnc(O)c1 c1(OC)cc(C)c(C(N2CC(CNC(c3cnsn3)=O)C(C)C2)=O)cc1OC Cc1cc2c(cc(C(=O)OCC(=O)CC3CCCS3)n2CC(F)(F)F)s1 c1(C(N2CC(NC(C(CC)n3cncn3)=O)C(C)C2)=O)cc([N+](=O)[O-])n[nH]1 CC(C)CC(O)C(=O)NC(C)(C(=O)NCC1(O)CC1)C1CCC1 c1(NC(C2C3(CN(Cc4ccc(C#N)cc4F)C3)C2)=O)c(F)c(F)nc(F)c1F N1(C(C(CCC)C)=O)CCC(CO)C(NC(=O)Cc2ccc(Cl)cn2)C1 C#CCC(CC(=O)NCC1(C#C)CCCC1)NC(=O)COc1ccsn1 C1(C(N2CC3C(NC(c4c[nH]c5nccc-5c4)=O)(C3)C2)=O)CCOCC12CCCCC2 C1(NC(=O)C#CC2CCCCC2)COC2(CCN(C(=O)CCC3CCC3)CC2)C1 c1(CC)ccc(C)cc1NC(=O)C(C(C)C)NC(C1(C#N)CCCOC1)=O C12(CNC(c3oc(C)c(Br)c3)=O)CCC(CC1)N2C(=O)C=C1CCOCC1 N1(C(COCC(=C)C)=O)CC2(CCN(C(=O)C(C)c3ccsn3)C2)C1 C(C)(C)(C(C)CC(=O)NCCc1ncccn1)NC(C(C)n1cccn1)=O c1(C(=O)NC(C(=O)NC(CC=C)C)C)cc2occc2[nH]1 C1(C(=O)NCCC)CCCN(C(c2ccn(C)c2CC(=O)O)=O)C1 N1(C(C2CCN(CC)CC2)=O)CC2CC(C(=O)NC3CCCCCC3F)(C2)C1 N1(C(=O)NCC2CCN(C(=O)OC(C)(C)C)C2)CCOC(C2CC2)CC1 N1(CC(C)N(C)C)CCC(C)(C(N2CCN(c3ccccc3)CC2)=O)CC1 CC(C(=O)NCCOCC(=O)NCC1(Cl)CC1(F)F)C(C)(C)C c1(C(C(=O)NC2(CCSCC(=O)NC3(CCCF)CCC3)CC2)=O)cccnc1 C1(NC(C2(n3cccn3)CCC2)=O)CCN(C(C2C3COCC23)=O)CC1O CCC(C)(CNC(=O)C(N1CCNC1=O)C)C(=O)NCCCCCCCO C(=O)(C1=CCCN(C(c2ccc3occc3c2)=O)C1)NC(c1ccc(C)nc1)C N1(C(CCC(=O)N(C)C)=O)CCC2(NC(=O)C=CCn3cncn3)CCCC12 O=C(C#CC1CCOCC1)NCC1CC(F)(F)CN1C(c1ccoc1Cl)=O N1(C(c2ccc(C(=O)O)cc2Cl)=O)CC2OCCN(C(C3CCCS3)=O)C2C1 c1(C(c2n(CC)nnn2)NCC2(C)CCOC2)cn(C)nc1-c1ccccc1 c1(NC2CCN(C(c3c(C)cc(C4CC4)nc3)=O)CC2C)ncnc2sccc12 CC1CCCCN1C(=O)CN1CCCC(CCNC(=O)CCn2ccnc2)C1 C1(C(=O)OC)CC2(CCNCC2)CN1C(=O)CN(C)C(N)=O C1(COC)(CNC(C2(C)CCOCC2)=O)CCCN1C(=O)CCc1ccc(C)o1 C1(C(=O)NC(C(=O)N(CCCC)CCO)CC2CCC2)CN2CCC1CC2 Cc1cc(C(N2CCC(NC(=O)COCC(F)F)C(CO)CC2)=O)cc(=O)n1C N1(c2nnc(COC)s2)C(CNC(=O)CC=C(C)C)CC2COCC12 c1(C(=O)NCCCC(C)NC(c2nnn(CC)c2C)=O)cc(C)c(C(F)F)cn1 C(=O)(C1CCCc2cc(C#N)ccc21)NC(c1ccc(C(C)C)cc1)CC(C)C Cc1cccc(C(N2CCCC2C(=O)NCCCC(=O)Nc2ccc(Br)cc2)=O)c1F C1(C(=O)NC(C)CN(C)C(c2csc(S)n2)=O)CCCCN1C(N)=O CC(CC(N)=O)C(=O)N1CCCC1C1(NC(c2cc3c([nH]2)CCC3)=O)CC1 C1(CC)(NC(c2nnnn2CC2CC2)CCC2OCCO2)CCCCC1 CC1CN(C(=O)Cc2cccc(F)c2O)CCCN1C(C1CC(=O)NC1(C)C)=O C1(C2(C(=O)OC(C)C(N3CCN(c4ccccn4)CC3)=O)CC2)NC(=O)NC1=O C1(O)(C(=O)NC(CCNC(CC(CC)C)=O)C)CCCC(C)(C)C1 c1(C(N(C(CCNC(c2ccc(C)[nH]2)=O)C)C)=O)csc2cncn12 C=CC1CN(C(=O)CCCCCOC)CC1NC(c1cc(F)c(OC)cc1N)=O N1(CC(=O)NCCCC(C)NC(C2CC(C3CC3)C2)=O)C(=O)NC(C)(C)C1=O O=C(CCCCC(F)F)NCCC1CC(F)(F)CN1C(c1cnc(S)[nH]1)=O Cc1cnn2c1CN(C(C1COCCN(c3nccnc3N(C)C)C1)=O)CC2 c1(SC)ncc(N)c(C(=O)NC(CO)C(C)NC(c2csc3cncn23)=O)n1 C1(C(=O)NCC(CC)NC(c2cccc(Cn3ccnn3)c2)=O)CC(F)CN1C C(C)(CCCN=c1[nH]cc2ncnc-2[nH]1)NC(CCCc1ccc(OC)cc1)=O CCCCC(F)C(=O)NCC1(CO)CCN(C(=O)C(C)N(C)C)C1 c1(C(=O)NCCC(C(C)C)NC(c2nn[nH]c2Cl)=O)ccc2c[nH]nc2c1 C1(NC(CC(C)OC)=O)C2CC1N(C(=O)CN1CCC(C)(O)C1)C2 N1(C(CC2CCC(OC)CC2)=O)CCCC2(C1)CN(C(C13CC(F)C1C3)=O)C2 C#CCCCC(C)C(=O)NCC(C1CC1)NC(c1cc(F)c(F)c(F)c1)=O N1(c2cc(CC)nc(CC)n2)CCC(C2(NC(=O)C3=CS(=O)CCC3)CC2)CC1 CC(CC1CC1)C(=O)NCCCOCCNC(=O)C(C)(C)c1nncn1C c1(C(=O)OCc2nnc(C3CCCC3)o2)ncn2c1CCCCC2 c1(C(=O)NCCN(CC(F)(F)F)C)nc(Br)n2c1CCC2 N1(C(CCc2n(C)ccn2)=O)CCOCC1CC(=O)NCCN1CCC(C)(C)C1 Cc1ccc(S(=O)(=O)C2CCCCC2NC(C2C=CCCC2)=O)cc1 N1(C(CSCC)=O)CC2(C(N3CCC4(C3)CN(C(C)=O)C4)=O)CC1CCO2 CC1(O)CCCC1n1cc(CCC(=O)NC2CCOCC2O)nn1 N1(C(C(CN(C)C)NC(C(CC)=CCCC)=O)=O)CCCC1(C)COC c1(NC(N)=O)ccc(Cl)c(C(N2CC(CNC(C3CC34CCC4)=O)C(O)C2)=O)c1 CC1CCCC(C)N1CCC(N1CCN(CCN(C(=O)C(=O)N(C)C)C)CC1)=O C1(C(C)NC(=O)C=CC(C)NC(=O)CCC(C)N(C)C)C(C)(C)C1(C)C C(CCC(CCC)NC(c1sccc1CC#N)=O)NC(CCSCCC)=O CCC(CC(=O)NCCOC1CN(C(=O)Cc2cc(=O)n(CC(C)C)[nH]2)C1)SC c1(CCC)[nH]nc2ccc(C(=O)NCCOCCCNC(C3CC3(F)Cl)=O)cc12 C(CN=c1[nH]c(N(CCCO)C)nc2c1CCCC2)c1cccc(OCC)n1 C(C(O)CC(=O)NC1CN(c2ncco2)C1)NC(C1(C)CCC1)=O c1(C(N2CC(C(C)NC(=O)C(c3ccccc3F)C)C2)=O)cnccc1Cl N1(C(c2cc(OCC)ncc2)=O)CCCC2C1CCCN2C(=O)Cn1cccn1 C12(CNC(C(C)c3ccsc3)=O)CN(C(C3C(C)(C)C3(C)C)=O)CC(F)(C1)C2 C1(C(N2CCC(NC(C(C)(C)SC)=O)C2C(C)C)=O)CCC2(CCC2)O1 C1(C(=O)C(F)(F)F)CCN(C(c2c[nH]nc2-c2ccc(F)cc2)=O)CC1 CCCCC(C(=O)N1CC=CC(NC(c2cc(CC)nc(O)c2)=O)C1)ON=C(C)C c1(C(N2CCC(NC(C3CC=C(C)CC3)=O)C2)=O)ccccc1S(=O)(=O)C(C)C C1(C(=O)NCCN(CC(C)O)C(c2c(C)csc2)=O)CC2(C1)CC(F)C2 C=CC1CCCN1CC(=O)NC1CCCC1Oc1ccccc1 Cc1ccc(CNC(C2(F)CCN(Cc3ccc(OC(C)C)cc3)C2)=O)c(O)c1 c1(CNC(C2OCCC(NC(C(CC)C)=O)C2)=O)cccc(F)c1C C(CCC)(C(O)C(=O)N(C)Cc1cn(CC)nn1)NC(C(C=C)(F)F)=O C(=O)(C1=CC2C=CC(C1)C2)N1CC(CNC(c2c(N(C)C)cccn2)=O)C(O)C1 CCCCCC(C)(C)C(=O)NCC(CC1CC1)C(=O)N1CCCC(N(C)C)C1 C(=O)(C(CC)OC)N(CCC(=O)NC1(C(=O)NCC#C)CC1)CCO c1(C(=O)NC(CC)CNC(=O)C=Cc2nccs2)ccc2c(c1)nc(O)n2C N1(CC(=C)Cl)C2CCC1CN(C(C1CCC(=O)N(CC)C1)=O)CC2 c1(N(C)C)cc(C(=O)NCC(C)(O)CNC(=O)C(C)(C)N2CCOCC2)nn1C N1(C(CN2CC(C)C2)=O)CCC(CNC(=O)CN2CCNC(=O)C2)C(C)C1 N1(C(C(C)SCC)=O)CCCC2(CCN(C(=O)C=Cc3ccc(Cl)cc3)C2)C1 n12cnc3c(nc(N4CC5CCC5(C)C4)nc13)N(C)C2.C1(CC)CCOCC1 c1(C(=O)NCC#CCNC(C(CC=CC)C)=O)c(C)[nH]c2ncccc12 c1(C(=O)NC(C23CCC(CC2)C3)CNC(C(COC)C)=O)ccnnc1O N1(C(COCCC#C)=O)CC2CCN(C(c3cc4nc(C)sc4[nH]3)=O)C2C1 c1(CN(C(=O)Cc2cn[nH]c2)C)ccc(CNC(c2ccc(Cl)s2)=O)cc1 N1(C(CCC=C)=O)CC(CNC(c2cccc(F)c2C(C)C)=O)C(F)(F)C1 N1(C(C(C)SC)=O)CCC(C)(CCNC(c2cc(F)c[nH]2)=O)C1 C1(CNC(c2ccnc3[nH]ncc23)=O)CN(C(C23CC(C2)C3)=O)CCC1(F)F C1(NC(c2cc(CC)no2)=O)CN(C(=O)C(C)CN(C)C)CC2CCCC12 c1(C(=O)NC2C(C)CCN(C(C=CC(n3cncn3)C)=O)C2)ncnc2c1CCC2 N1(C(c2ccc(NC)cc2)=O)CCC2C(C(=O)NCCC3(COC)CC3)C2C1 CCC1=NOC(C(=O)N(C2(C(=O)NCC(F)Br)CC2)C)C1 C(=O)(CC(O)CC(C)C)N1C(CNC(=O)C(O)C2CC2)CC(OC)C1 CCCCC(CNC(=O)C=CS(C)=O)NC(=O)C(c1cccc(F)c1)(C)C c1(CC)cc(N2CCC(NC(c3cn(C(C)C)nc3C)=O)C(C)C2)nc(C)n1 CC(C)C(C)(O)C(=O)N1CC(C(C)(C)O)(CNC(c2c[nH]cc(F)c2=O)=O)C1 Cc1cc(C(=O)NC2CC(F)(F)CC2NC(c2cnns2)=O)c2ccccc2n1 c1(C(N2CCCC(F)(CO)C2)C(=O)NCC(=C)C)nc2c(s1)CC(C)(C)CC2 C1(O)(CNC(CCC=CC(C)C)=O)CCCN(C(=O)C(C)(C)OC(C)C)C1 C1(CCNC(C(C2CCC2)COCC)=O)(OC)CN(C(=O)CCNC(=O)C=CCl)C1 c1(C(N(CCCN(C)C)CCNC(C2CC2(C)C)=O)=O)cn2cccc(F)c2n1 CCCCC(O)C(C)C(=O)N1CCC(NC(c2cc(O)cs2)=O)C1 S(=O)(=O)(c1ccc(NCCCOCC)c(C#N)c1)N(C(CCOC)C)C c1(C(=O)OC)cc(C(=O)NC23CC(CNC(=O)CN4CCCC4=O)(C2)C3)cn1C c1(C(=O)NC(C)CCCNC(=O)C(C)Cn2ccnc2)ncc(F)cc1N CC(C(C(=O)NC1CCC1)N1CCCC1C(N1CCCC1)=O)C1CC1 Fc1cc(Br)cc(CNC23CCCCC2C3)c1F C1(C(=O)Nc2cccc(NC=O)c2)CC2CC1CC2NC(=O)C(O)c1ccco1 Cc1ccc(C(=O)NC2CCCC2(C)CNC(c2nsnc2O)=O)cc1C C1(NC(C(C)(O)C2CCC2)=O)CC(F)CN(C(c2sccc2SC(F)F)=O)C1 C(=O)(CCCC(F)(F)F)NC(CCN(C)C)C(N1CCC(=C(F)F)CC1)=O C1(CC=C)(NC(C2CCN(c3ncc(OCC)cn3)CC2)=O)CCOCC1 CCCS(=O)(=O)C(C)C(=O)N1CC2CC2(CNC(C2(C#N)CCSCC2)=O)C1 N1(C(c2c[nH]nc2Br)=O)C2CCC1CC(n1cc(C3OCCO3)nn1)C2 Cn1cc2cccc(C(=O)NC3CC3CNC(c3cccc(N)n3)=O)c2n1 CC1CCC=C1C(=O)N1CCN(C(c2cc(=O)c(Br)c[nH]2)=O)C(CCO)C1 Cc1c(C(=O)NC(CCN(C)C(C2CC(=O)NC2(C)C)=O)C(C)C)cccc1O C(N=c1nc2c(cnn2C)c(NC2CCOCC2F)[nH]1)c1c(CC)n[nH]c1 C(=O)(CCCS(C)(=O)=O)N1CC(CNC(c2c(CC)n(C)cc2)=O)OCCC1 CS(=O)(=O)c1ccccc1CNC(C1(F)CCN(C(=O)Cc2ccccn2)C1)=O C1(N(C(=O)CCOC2CC2)C)CCCN(C(=O)Cn2cc(C(F)(F)F)nn2)C1 c1(-n2c(C)ncc2)ccc(C(=O)NCC(O)CNC(C2(F)CC2C)=O)cn1 C1(CC(=O)OC)CN(CC(C)CC2CCC2)CC(C)(C)O1 c1(-c2cn(-c3c(CC(=O)O)cccc3)nn2)cnc(CCNC(=O)CSC)nc1O CC1=C(C(=O)NC23CN(C(=O)CC(C)C(C)C(C)C)C2C3CC)C(C)(C)CCC1 C=C(C)C1OCCCC1C(=O)NCCCCN(C)C(C1CCCCC1CC)=O C1(CC(=O)NC2C(NC(C3(C=C)CCC3)=O)CCCC2)CN2CCN1CC2 C(=O)(C1CCSc2ccccc21)N(CC(C)NC(C1CCN(CC)CC1)=O)C N1(C(c2c(C)nn(CC(F)F)c2)=O)CCC(O)c2cc(Br)ccc2C1 C#CCC(C)C(=O)N1CCC(N(CC)NC(C2COCCN2CC)=O)C1 N1(C(C(CCN(C)C)NC(=O)CCN2CCCC2=O)=O)CC(S(C)(=N)=O)C1 c1(C(N(C2CCN(C(CC(C)F)=O)C2)CC2CC2)=O)cccc(Cl)c1 N1(C(CC2(OC)CCCC2)=O)CCCC(CCNC(=O)C(O)C(C)C)C1 C1(NC(CC(C)SC)=O)CCC(CNC(=O)Cn2cc(C3CC3)cn2)CC1 N1(C(=O)NCC2C(C(=O)OC)C2)CCCC2(CCCO2)CC1 CN1CC2CC1CN(C(c1ccc(C(F)(F)F)cn1)C(=O)NC1CCC1)C2 C1(C)(CNC(CCC=CC)=O)CCCN1C(C1CC1c1ccncc1)=O N#Cc1c(N2CCC3(CC2)CC3C(=O)NC2CCCC2C2CC2)cccc1F c1(NC(c2n(CC)nnn2)c2ccc(COC)s2)cccc(CCC(N)=O)c1 C(=O)(C(CCOC)OC)NC(C(=O)NC(C=C)(C)C)C1(O)CCC1 C1(NC(C2N(C(C3C(C)CCOC3)=O)CC2)=O)CCC(C2CC2)C1 C=C=CC(C)C(=O)NCC1(OC)CCN(C(c2cc(CC(C)C)nn2C)=O)C1 c1(CC)[nH]ccc1C(=O)NCCCC1CCCN1C(C1CSCCS1)=O CCC(C#N)C(=O)N1CCC(N2CCN(C(=O)Cc3csc(S)n3)CC2)C1 N1(c2ccnc(OC)n2)CCC(NC(=O)CCN2CCOCC2)C(F)C1 c1(C(=O)NCC(C)NC(=O)C(O)C2CC2)c[nH]c(C(F)(F)F)c1 Fc1ccc(N2CCOCC2CCNCC2C=CCC2)cc1 c1(C(N2CCC(N(C(C3CC(SC)C3)=O)C)CC2)=O)c(F)ccc2c1OCC2 C1(C(=O)NCC2C(C)=NNC2=O)CC2(CC(NC(=O)C(C)NC=O)C2)C1 C12(C(=O)NCC3CN(C(C(C4CC=C(C)CC4)F)=O)CC3O)CCN(CC1)CC2 C1(CNC(C=CC)=O)CN(C(C2CCC2(OC)OC)=O)CC12CC2 C=CCC(C)(C)CC(=O)NC1CC(CNC(c2cc(CC)no2)=O)C(O)C1 C1(NC(c2c(CC)noc2C)=O)CN(C(=O)C=Cc2cncn2C)CCC1C C(=O)(C(F)(F)C(F)(F)Cl)OCC(c1cn(C2CCCN(CC)C2)nn1)(C)O C(CCC(C(=O)Nc1cccc(C(C)=O)c1)NC(C1CCOC(=O)CC1)=O)OC N1(C(C(C)=CC2CC2)=O)CC(N(C(=O)CCC2CCCCO2)C)C(C)(C)C1 C1(C)(C(=O)NC2CC(CCNC(CN(S(C)(=O)=O)C)=O)C2)CCCC1 Cc1cc(-c2nn[nH]n2)c2sc(C(=O)N=c3nc[nH]s3)cc2n1 n1(C(C2CCOCC2)C)nc(-c2ccccc2)nc1C1CCC1(F)F c1(C(=O)NC2CN(C(=O)CCC3CCCC3)C2)c(Cl)cccc1Br CC(C)C(C)(CNC(=O)CCOC1CC1)NC(c1ccc(CO)cn1)=O CC(C)(C)CC(O)C(=O)NC(C)(C)CC(F)C(=O)N1CCCC(C)(CO)C1 C1(CC(=O)NCCN(C(=O)CCc2ccc(C)s2)CC)COCCN1CC C1(C(=O)NC2CN(C(=O)OC)C2)CCCN(C(=O)Cn2ccnn2)C1C C1(NC(c2scc(C)c2)=O)CCN(C(c2ccc(C(O)CF)cc2)=O)C1(C)C N1(C(CNC(CC)=O)=O)C2CCC1C(NC(=O)C(F)n1ccnc1)C2 N1(C(C(CN(C(c2cncc(C)c2)=O)C)C)=O)CC2CCC(CC2)C1 C1(N(C)C)CCCN(C(C2COCC2NC(C2CCCCO2)=O)=O)C1 N1(C(CCSCCC)=O)CC(C)(C)CC1C(=O)NC1CN(C)CC1(C)C C1(CNC(=O)CCc2cnoc2)CCCC(NC(=O)C(C2CCOCC2)O)C1 c1(C(N2CC3(CC(CNC(C(C=C)O)=O)OC3)C2)=O)cnc2c(c1)NC(=O)CN2 N1(C(CCCCOC)=O)CCC2CCCC12CNC(=O)CCCC(=O)N(C)C CCC1(CC)CN(C(C)=O)c2ccccc21.C12CC(C1)OC(=O)C2 Cc1ccc(SCC(=O)NC2CN(C(=O)CC3CC=CCC3)C(C)(C)C2)cc1C CC1CN(C(c2ccn(C3CCC3)n2)=O)CCC1NC(=O)Cc1nnc(O)s1 c1(C(=O)NCc2c(C)cc(-c3nn[nH]n3)cc2)nnc2cc(C#N)ccn12 C12(C(=O)NC(CC)CNC(c3cc(=O)cc[nH]3)=O)CCC(CC1(F)F)C2 c1(C(=O)NC(CCCNC(C(N2CCNC2=O)C)=O)(C)C)cnn2c1N(C)CC2 c1(C(=O)NCCn2cc(-c3cccs3)nn2)ccc(CN2CCC(O)CC2)cc1 N1(C(c2c(CC)nccn2)=O)CCC(CNC(C2CCCSC2)=O)C12CCC2 C(=O)(C(C(C)(C)C)OC)NCCC(C)(C)NC(C(CC)CC1CCCCC1)=O c1(CC(=O)NC2CC(F)(CNC(C(CC)=CC)=O)C2)sc(-c2ccsc2)nc1C O=c1c2ccccc2ncn1Cc1nc(-c2nc(C(F)(F)F)cs2)nn1C1CC1 c1(C(=O)NCCCN(C)C(C2CCCOC2)=O)cc(N2CCCC2)ccn1 CC(CCN=c1[nH]c(N(C)Cc2cccn2C)nc2c1COC2)CC(C)(C)C CCC(C)(CNC(=O)C(O)C1CC1)NC(c1cc(Cc2ccccc2)c[nH]1)=O N(C1CCCn2nccc21)C(c1nnnn1C1(C)CC1)(COC(C)C)C C(=O)(CS(=O)(=O)C(C)(C)C)NC1(COC)CCN(C(=O)CC2(O)CCCC2)C1 C#CC1CC2(CC(C(=O)NCCN(C(=O)CCN3CCCC3)CC(C)O)C2)C1 N1(C(CNS(CC)(=O)=O)=O)CC2CN(C(c3cnn(C(C)C)c3C)=O)CC2(C)C1 C#CCCCCC(=O)NCC(=O)NC1CCCC12CC2 CC1C(C(=O)NCCc2c[nH]nc2O)CCN1C(=O)C(C1CCCCC1)=O c1(CCC)sc(C(=O)N(CCCNC(=O)CC(C)F)C2CC2)cc1Br C1(C(N(C(C)(C)CC(N2CCC(C)(CO)C2)=O)C)=O)CCCC2(CC2)C1 c1(OCCC)ccc(NC(c2cc(C(C)C)n(C(C)(C)C)n2)=O)cc1C CC1(C)CN(C(=O)C2=NOC(C)(C)C2)C(CNC(c2ccc(Cl)cn2)=O)CO1 CC(C)(C#N)CC(=O)N1CC(O)(CNC(c2cc(F)cc(Cl)c2)=O)C1 C(=O)(C1=CC2(CCN(C(C3CC4(CC4)C3)=O)C2)C1)NCCCCC#C Cc1ncc(N)cc1C(=O)NCCC1CCN(C(=O)C(C)C(F)F)C1 C1(C(=O)NCCN(C(CC2CCN(C)C2)=O)C2CC2)CCCNS1(=O)=O S(=O)(=O)(c1ccc(NCC2CSCCS2)c(C#N)c1)N1Cc2c(nc(C)s2)CC1 CCCC(C(=O)NCC1CC(NC(C2CC(F)(F)CC2C(=O)OC)=O)C1)C(C)C C(=O)(C(O)CC(F)F)N1CC(C(C)NC(C2CC2[N+](=O)[O-])=O)C1 N1(C(C23CC(NC(C(COC)OC)=O)(C2)C3)=O)CCC(CO)C(O)C1 N1(C(C(C)OCc2ccc(N(C)C)cc2)=O)CC2(CCN2C(C2CC2(F)F)=O)C1 N1(CC2(OCC)CCCOC2)CCC2(CCCC2)CC1 Cc1ccnc(C)c1C(=O)NCCC(O)CNC(c1cn(C)c(=O)cn1)=O C1(NC(CSCC#C)=O)CC(CC(=O)N(CCCC)CCO)C1 c1(C(=O)NC2CN(C(CCCC)=O)CC2c2ccc(F)cc2)cc(Cl)cnc1O N1(CCCCNC(CNC(C)=O)=O)CCCN(C(C23CCCC2C3(F)F)=O)CC1 C#CC1(NC(c2ccc(SCc3ccco3)cc2)=O)CCC(C)(C)C1 C1(NC(c2cc(OC)no2)=O)C2CCC(C2)C1C(N1CCCCC1CC(C)C)=O C=CC(C)CC(=O)N1CCC1C(=O)NC(C)C(C)SC Cc1ccc(CCNC(c2ccc(-c3cn[nH]c3)cn2)=O)cc1 c1(CC(=O)NC2CCC2c2cccc(-c3nn[nH]n3)c2)cccc(F)c1F Cc1cnccc1CN(C(C1CCCCC1)C(=O)NCCC#N)C C1(CNC(CNC(c2c(C)occ2)=O)=O)CCC(C)N(C(=O)CC2CC=CC2)C1 c1(COC)nc(=NC2(CNC(c3c(C)ccnc3Cl)=O)CCCCCC2)s[nH]1 CC(C)CC(C(=O)N1CC(CCNC(=O)C(C)N(C)C)C1)c1ccccc1 C1(C(N(C)CC2CN(C(C3CCC3)=O)CCO2)=O)CS(=O)(=O)CC12CC2 c1(C(=O)NC2CC3(CC(NC(c4c(C)scn4)=O)C3)C2)ccnc2c1ncn2C c1(CC)cc(N2CCN(CC)CC2)ccc1F.c12cn(nn1)C(C)C(=O)NC2 CC(CS(=O)(=O)N1CCC(NCc2ccc(Cl)cc2F)CC1)C(=O)O N1(C(C2CC(OC)C2)=O)CC(NC(=O)COc2cc(C)ccc2F)CC1(C)C Nc1c(C(=O)NCc2ncccc2CNC(C2CCN2)=O)ccc(Cl)c1F c1(Cn2cc(NC(C)=O)nn2)ncc(Br)cc1OC.c12n[nH]c(c1C)C(=O)NO2.CO c1(CC)[nH]nc(C(=O)NCC2CC2NC(C2CCCN2C(C)=O)=O)c1Cl c1(C(N2CCCC(C)C2)C(=O)Nc2c(C)cccc2C)cc(F)c(Cl)cc1Cl N1(C(c2ccc(C)cc2Br)=O)CCCC2CN(C(=O)C(C)(C)CO)CCC12 N1(C(CN(C(C2C(C)SCCC2)=O)C)=O)CCC2(C1)CN(C)C2 CCC(CC)CCCC(=O)N1CCN(C(=O)CCCNC(C)=O)C(C2CCC2)C1 C1(CCNC(C2CC(C3CC3)=NO2)=O)CN(C(C2(F)CC2)=O)CCS1(=O)=O c12cncc(c1)c1csc(c1)c2=O.C1(N(C)C(=O)O)CC1(C)C CCCC(C)(C)C(=O)NCC(CCOC)NC(=O)CNC(c1ccc(C)cc1)=O c1(CC)ccc(F)c(C(N2CCC(NC(C3(F)CCOC3)=O)C(O)C2)=O)c1 N1(C(C(C)NC(=O)CCc2ccsc2)=O)CCCC(CCN(S(CC)(=O)=O)C)C1 C(C(=O)NOCC1CCC1)(NC(C(COC)OC)=O)SC N1(C(C(C=C)(C)O)=O)C2CCC1(CNC(c1scnc1COC)=O)CC2 C1(NC(CS(=O)(=O)NC)=O)COCCN(C(c2cnc(C(F)(F)F)s2)=O)C1 CCC(CCCC(=O)N(C1CCCCC1)CC1CC1)NC(=O)C(C)N(C)CC CC(CC(F)(F)F)C(=O)NC1(CNC(c2nc[nH]c3nccc2-3)=O)CCOC1 c1(C(C)NC(C(F)=CC)=O)ccc(CNC(c2cnn(C3CCC3)c2C)=O)cc1 C1(CNC(=O)NC(c2cnc(C)s2)C)CCc2nn(C)cc2C1 c1(CN2CC(NC(c3cc(F)ccc3C(F)(F)F)=O)C2)cc(Br)cc2[nH]ccc12 c1(-n2cc(CNC)nn2)ccc2c(c1)CN(C(c1cc(F)c(Cl)c(Br)c1)=O)CC2 C1(C(N(C(CC#C)C)C)=O)CC2CCCC2N1C(C1CCC2CC1CO2)=O n1(CC(=O)NC2C(NC(c3c(C)n(CCO)cc3)=O)CC2)c([N+](=O)[O-])cnc1C c1(C(=O)NCC23OCCC(NC(C4(C)CC4)=O)(C2)C3)cncc2c1CCNC2=O C(N=c1nc(N2CCC(C)(CO)C2)c2c([nH]1)CSC2)c1n(C)cnn1 N1(C(c2cc(C)nc(C)c2)=O)CCC2(CC1)CC(C(=O)NCC1CC1)CO2 C1(CCNC(C(C)NC(COC)=O)=O)CCCCN1C(C1(c2cc[nH]n2)CC1)=O c1(NC(C(CCSCC)NC(=O)CC2COCCOC2)=O)cc(CC)cc(O)c1 C(CCC(O)C(=O)NCC#CC(F)(F)F)NC(C1CC(O)C(F)C1)=O c1(C(=O)NCC2CCN(C(c3ccc(OC)cc3Cl)=O)C2)cc2sc(C)cc2s1 C=CC1OCCC1C(=O)N(CCNC(=O)C(c1cccnc1)OC)C1CC1 Cc1ncnc(NCC2(NC(=O)CC(C)C3CCCO3)CCCCC2C)c1C#N c1(OC)ccc(-c2cc(CN=C(NC3CCOCC3)NC3CCC3)no2)cc1 n1(C(C)C)cc(OCC(=O)NC2CC(NC(=O)CC3CNC(=O)O3)C2)cn1 c1(C(N2CC(O)(CCNC(CC3CCC(C)CO3)=O)C2)=O)cc2ccccc2[nH]1 C1(C(=O)NC(=O)CNCCN(CCN(CC(C)O)CC)CC)CCCCC1C1CC1 c1(SC)ccc(CC(=O)Nc2ccc(OCF)cc2)cn1 C1(C)(CNC(C2C3(CC(OCC)C3)C2)=O)CC(F)(F)CN1C(=O)CC1(C)CCC1 c1(C(CC)C)ccc(C(=O)NCC2(F)CC(CNC(C3CC(C)(F)C3)=O)C2)cc1 c1(OCC#C)ncccc1C(N1CCC(C(C)NC(c2coc(CC)n2)=O)C1)=O C(=O)(C1CCCn2nccc21)N(C)CC1(NC(C(C(F)(F)F)OC(C)=O)=O)CC1 C1(NC(c2c(C)cns2)=O)CCN(c2cc(OC(C)C)ncn2)CC(C)(C)C1 N1(CC(=O)N(C)C)CCCC(CN=C(NCC(C)(C)C)NC2(CO)CCCC2)C1 C(CCCCCCC(=O)N1CCC(NC(c2cc(C)ncn2)=O)C12CCC2)SC N1(Cc2scc(C(=O)OC)n2)CCC(C(C)C(=O)Nc2csc(SC)c2)CC1 N1(C(=O)CC2CCC2NC(=O)CCc2cncnc2)CCC(F)(F)CC1 c1(C(C(=O)Nc2c(C)cccc2)N(C2CCC2)C2CC2)c2c(nn1C)CCCC2 C(=O)(C1CCCc2nncn21)N(CCN(C(=O)CNS(N)(=O)=O)C(C)C)C c1(C(=O)NC(C)CC2CN(C(c3ccnn3C3CC3)=O)C2)cc(Br)n(C)c1 CC1C(NC(C2CCS(=O)(=O)N2)=O)CCN1C(=O)CCc1ccc(N(C)C)cc1 C1(C(N2C(C(=O)NCC3CC(CN=[N+]=[N-])C3)CC2)=O)CC2CCC1C2 c1(OC)nc(N(c2ccccc2)C2CC2)ncc1C.N12CCCCC1C2=O C1(OC)CCC(C(=O)NCc2cc(C(=O)NCc3nnn(C)n3)n[nH]2)CC1 N1(C(C2N(C(C3CCC(=O)C3)=O)C3CCC2C3)=O)CCn2ccnc2C1 Cc1cc2ccccc2nc1C(=O)NCCCNC(=O)C(F)(F)c1nccn1C c1(COC2CN(C3(C)CC3)C2)nocc1C(=O)NC.C1(=O)CCN1.C1CCCO1 Cc1nc(=N)[nH]cc1C(=O)NCCOC1CCN(C(c2cncnc2)=O)CC1 C1(C(N2C(C(N(CC#C)CCF)=O)C=CC2)=O)C2CC(=O)CC12 O=C(C#CC1CCOCC1)NCC(CC1CCCC1)C(=O)NCC1CCSC1 S(=O)(=O)(c1ccc(Cl)c([N+](=O)[O-])c1)N1CCC(NS(c2ccn(C)n2)(=O)=O)C1 c1(C(=O)OC)cc(CCNC(=O)CNC(=O)NC(c2cc(C)on2)C)on1 c1(C(N2C(CNC(C3(COC)CCOC3)=O)CC2)=O)c(C)oc(C)c1S(N)(=O)=O N1(C(C(CCCC)NC(c2nnsc2N)=O)=O)C2C=CCC1CCC2 c1(C(N2CCC(O)(CCNC(C3ON=C(C)C3)=O)C2)=O)cncc(Br)c1C Cc1ccc(C(N2CCOCC(NC(C3C=CCCC3)=O)C2)=O)c(O)c1C c1(C(=O)NCC(CNC(CC(CC)C2CC2)=O)O)[nH]c2ccccc2c1Cl N1(C(C=CSC)=O)CCC2(CCCCC2NC(c2ccsc2C(F)F)=O)C1 C(C(C)(O)CC(=O)N1CCC(C(=O)NC2(C(O)CO)CC2)C(C)C1)OC C1(N=[N+]=[N-])(C(=O)NCC2C(C)NC(=O)CC2)CCN(C(C2CCN2C)=O)C1 C1(CCNC(CCC(=O)OCC)=O)CCN(C(=O)Cc2cnc(C)[nH]2)C(C)C1 C1(C(=O)NCC2CCN(CCN(C)C)CC2)C(N)C2CCCC12 C1(CC=C)(C(=O)NCC(CC)NC(=O)COC2CC=CC2)CCOCC1 C1(CNC(=O)CCOCC2CCC2)CC2CCCC2N1C(=O)C=Cc1ccc[nH]1 C(=O)(CCCCCC(C)O)NC1(CNC(C(CC)n2cccn2)=O)CCCCC1 Cc1c(CN2CCC3(CC3C(=O)Nc3nccc(I)n3)C2)ccc(F)c1F CC(C)C(C)C(=O)NC1CC1CNC(=O)Cc1csc(-c2cccc(Cl)c2)n1 C1(O)(CC(N2CC(CNC(CC(C)C3CCCO3)=O)OCC2)=O)CCCN(C)C1 c1(-c2c(C(=O)NC3CC(NC(CCOCCC)=O)C3)con2)ccccc1Cl C1(C)(C(=O)NCC2CCC(NC(C=Cc3n(C)ncc3)=O)C2)CC(C2CC2)=NO1 C(=O)(CC1=CCCC1)NCC(CNC(C1(CC=C)CCOCC1)=O)C C1(C(CNC(c2cc(OC)no2)=O)C)CCN(C(c2cnn(C(C)C)n2)=O)CC1 C(=O)(C(C(C)C)c1cccnc1)NC1(CO)CN(C(CC(C)C)=O)C1 CCCCC(O)CC(=O)N1CC(O)CC1C(=O)N(C)Cc1cocn1 c1(C(N(CCn2cc(CNC3CCCNC3)nn2)CC)=O)cccc2c1OCC2C c1(NC(C(C)N(CC)CC)=O)cccc(NC(=O)CC2(C)CC2)c1 CCCC(CC)CCC(=O)N1CC2CC(C(N3CCC(O)CC3CC)=O)CC2C1 C1(CCCNC(c2c(CC)csc2)=O)CCCCN1C(=O)Cc1c(C)cnn1C N1(C(CC(C)C(C)(C)C)=O)CCC(C2CC2NC(c2ccc(CO)nc2)=O)CC1 c1(CC)cn2c(C(=O)NC3CC(C)(NC(c4cnco4)=O)C3)cccc2n1 Cc1cc(C(=O)OCC(c2cn[nH]c2)=O)c(C)n1CC1CCCOC1 CC#CCCCC(=O)NC1C=CC(CNC(=O)COCC(N2CCCC2)C)C1 C(=O)(C(C)(C)S(C)(=O)=O)NCC12C(CN(C(C3(C(C)C)CNC(=O)C3)=O)C1)CC2 Cc1[nH]c(C#N)cc1C(=O)NC1(C)CCCCC1C(N1CC2CC=CC1C2)=O C1(C)(OC)CCCN(c2nc(N3CCCC(C(F)(F)C(F)(F)F)C3)cc(C)n2)C1 N1(C(c2nn(CC)c(C)c2)=O)CCC2(CC1)CC2NC(=O)CN1CCCC1CO C(C)(C(=O)NCC1(CCNC(=O)C(C)OC2CCCC2)CC1)NC(C)=O S(=O)(=O)(c1ccccc1Cl)N1CCCC(CC(=O)NC2CCC(O)CC2)C1 N(C1COc2ccccc21)C(C1N(C(C=Cc2ccc(C)o2)=O)CCSC1)=O N1(C(C(N2CCC(O)CC2)C)=O)CCC2(CC1)CN(C(=O)Cn1nccn1)C2 c1(C(=O)NCC(CN(C(CSCC(=O)OC)=O)C)C)cc(C)c2c(O)n[nH]c2n1 C1(CC)CCN(C(=O)C(C)Cc2ccoc2)C1C(=O)NCC1CC2(CC2)C1 c1(C(N(C2CCC(NC(c3ccc(F)s3)=O)C2)C)=O)ccc2nc[nH]c2c1 C(CCC(C)(C)NC(C1CC1C(F)(F)F)=O)NC(CC1C(CC)C1)=O c1(C(=O)NC2CC(CNC(C(CSC)O)=O)C2)ccnc2ccc(Cl)cc12 CCCCCC(O)CC(=O)NC1CCN(C(=O)Cn2cnc([N+](=O)[O-])n2)C1C C1(CC(=O)N(C(C)C)C)CCCCC1NC(=O)C=Cc1nccs1 C(C(CC(C)C)C(=O)NCCCC(CO)NC(=O)C(C1CCCCC1)C)OC C1(Cl)(C(N2CC(OCCNC(CC3C(C)C3)=O)C2)=O)C2CCC(=O)C12 C1(CCCC)CN(C(c2cc(C)c(C)[nH]2)=O)CCN1C(C1C2COCC12)=O c1(C(N(C(CCNC(CCC(=C)Cl)=O)C)C)=O)cc(C#N)c2n1CCCC2 N1(C(CNS(CC)(=O)=O)=O)CC2(CC2)CC1CNC(=O)CN(C)C(=O)NC C1(C(N(CCN(C(C(COC)(C)O)=O)C)C(C)C)=O)CCCCS1(=O)=O c1(C(=O)OC)cn(CC(=O)NCC2CCC(NC(=O)CNC=O)C2)cn1 N1(C(C2C=CCCN2C(=O)Cc2ccns2)=O)CCCN2CCCC2C1 c1(C(=O)NC2C(NC(CCCCC=C)=O)C2)ccc(Cl)c(C)c1O O=C(C1=CC2(CCOC2)C1)NC1CN(C(=O)CCSc2ccccc2Cl)C1 CCC(C)C(CC(=O)NC(C)CCN(C)C)NC(=O)CC1C=NN(C)C1=O CC1C(=O)N(C)CCN1C(=O)COC1(C)CN(C(=O)C=Cc2cc[nH]c2)C1 c1(CN2C(C(=O)NC(C)CN(C)C)CSCC2)c[nH]c2ccccc12 c1(C(N2CC3C(C(N4CC(C)NC(=O)C4)=O)(C3)C2)=O)cc(F)ccc1C#N CCC(CCCC(=O)N1CC(c2ccncc2)C1)NC(C1CCN(OC)CC1)=O c1(C(=O)NC(C(C)C)CCN(C)C(C2(O)CCSCC2)=O)c(Cl)ccnc1F C(=O)(CCCCCn1cnnn1)NCC(C(C)(C)C)NC(=O)COCC1CCCO1 c1(C(=O)NCC(CNC(CCCC=C)=O)C)ccc(C)cc1Br c1(C(=O)NCCOCCCNC(=O)CC2CC=CCO2)ccc2ccncc2c1 N1(CC(=O)N(C(C2CC23CC3)=O)Cc2ccccc2Cl)CCN(c2ncccn2)CC1 N1(C(CCc2c(C)cccc2)=O)CC(NC(=O)C(O)c2cnc[nH]2)CC(F)C1 CC(CC1CCCO1)C(=O)NCCC1CC(NC(=O)CCC2(C)CC2)C1 N1(C(C(C)(C)OC)=O)CC2CCOCC2(NC(c2cc(C(C)=O)cn2C)=O)C1 N1(C(C(C)CC(N)=O)=O)CC2(CCOCC2)C1c1cn(CC2CCCO2)nn1 N1(C(c2ccc(N3CCCCC3)nc2)C(=O)NCC)CCOC2CS(=O)(=O)CC12 C1(NC(=O)OCC)C2CC3C1C3C2C(=O)NCCOC(F)F.C1C(=O)N1 C#CCN(OC)C(=O)C1C2CCN(C(c3cc[nH]c3CC)=O)CC12 C12(NC(CCN(CC)CC)=O)CCCCC1N(C(=O)C(c1ccccc1)=O)CC2 C(=O)(CC(CNC(=O)C(O)CSC)OC)NCC(CC)(C)O Cc1n[nH]c(C)c1S(=O)(=O)N1CCC(O)C(Nc2ncnc3ccccc23)C1 N1(C(c2cc(CC)on2)=O)CC2CC2(CNC(=O)C2=C(Cl)CC2)C1 CCCC(C)C(=O)NC1CN(C(=O)Cc2ccnc(OC)c2)CC1C C(=O)(CCP(C)(C)=O)NC1C(C)CN(C(c2cc(-c3ccc(Cl)cc3)no2)=O)C1 C12(CNC(c3cc(C#N)[nH]c3)=O)CN(C(=O)CC3CCOC3)CC1CS(=O)(=O)C2 c1(NC(C2CC(O)CN2C(=O)Cc2ccc(O)cc2)=O)c(F)ccc(Cl)c1F C1(NC(CNC(C)=O)=O)CCN(C(C2CCCN2C(=O)C(C)C)=O)CC1O c1(OC)cnccc1C(=O)NC(C)CC1CN(C(=O)CC(C)n2cccn2)C1 C1(CC(N2C(CC)CC2)=O)C=CC(NC(=O)C(CO)NC(N)=O)C1 C1(N(CCc2c(C)ccnc2)C)CCc2cc(Br)ccc2C1 c1(C(N2C(C)(C)C(CNC(C3OCC3(C)C)=O)CC2)=O)cccc(S(N)(=O)=O)c1 C(C(CC(C)C)C(=O)NC1CC12CC(NC(c1cccc3[nH]ncc13)=O)C2)OC c1(C(N2CCCC(O)(C3CC3)C2)C(=O)NCC(C)C)ccc2ccccc2n1 c1(C(=O)NCC(=O)NCCC(c2ccccc2)C)c[nH]c2cccnc12 N1(C(c2c(C)ncnc2C)=O)CCC2(CCCCC2NC(=O)CNS(N)(=O)=O)C1 C1(CCC)(NC(c2nc(CC)oc2C)=O)CCN(C(c2ccc(CC)o2)=O)CC1 C(=O)(C1=CCCCO1)N(C(CCNC(C(CC)NC(c1ccccc1)=O)=O)C)C Cc1cc(C(N2CC(NC(=O)CCCCBr)C(F)C2)=O)nn1C C1(CNC(=O)CC2COCCO2)CC(O)CN1C(c1cc(CCO)on1)=O CC(C)C(F)C(=O)NC(C)(C)C(=O)NCC1C(C)C1(F)F c1(C(=O)NC2CCC(N(C(=O)CN3CC(C)(C)C3)C)C2)nn(C)c2c1CCC2 C1(C(N(C2CCS(=O)(=O)C2)CC(CC)OC)=O)CCCCC1C(C)(C)C N1(C(c2cnn(C)c2C#N)=O)CC=C(CC(=O)NC2CCOC2(C)C)CC1 c1(CNC2CC(NC(CCC3CCC(C)O3)=O)C2)ncccc1Cl C1(C)(C(N(CC(O)CNC(C2(C3CCCO3)CCC2)=O)C)=O)CCCN1C N1(C(CC2(COC)CCOCC2)=O)CC(C)(C)CC1CNC(c1n[nH]cc1F)=O c1(OC)ccc(C(N2CC(OC)C(NC(C3CCN3C3CCCC3)=O)C2)=O)cc1 C=CCC(CC)C(=O)NCCOCCNC(=O)Cc1c(C)ncnc1C C(=O)(C(C)CC(C)C(C)=O)NCC(CC(=O)NC(CC)CCO)O C=CCC(C(=O)NC(C)C(C)NC(C1CCC(CCC)CC1)=O)C(C)C C(C)(CCCCN=c1[nH]cncc1I)NC(C1CC2CC(OC)CC21)=O N1(C(c2ccc(C(C)=O)o2)=O)CCC(C)(C)C(NC(c2cnc(O)cc2C)=O)C1 C1(NC(=O)C2=CCSC2)CC2CC(NC(C3CCCCNC3=O)=O)CC12 C1(CC(=O)N(CCNC(C23CC(OC)C2C3)=O)C)CCC2(CCCC2)CC1 Cc1ccc(NC(=O)CN(C)C(C2COC(C)C2)=O)c(C)c1 c1(C(N(C(C=C)C)C)=O)ccc(CNC(=O)CCn2cnc(=N)[nH]2)nc1 c1(-n2cc(CC(C(=O)NCCCOCC)O)nn2)c(F)cccc1[N+](=O)[O-] O(N1CCC(CC(N2CCCC(N(C(=O)C(C#N)CC)C)C2)=O)CC1)CC C1(O)(CNC(c2c[nH]nc2F)=O)CC(NC(C2(CC3CC3)CC2)=O)C1 C1(C(=O)O)CC(F)CN1C(=O)NC(c1ccc(Br)cn1)c1ccccc1 N1(C(c2snc(C)c2N)=O)CCC(NC(c2ccc(F)c(Cl)n2)=O)C(F)C1 C1(NC(CSCC(=O)OC)=O)CC(F)(F)CC1NC(c1ccnc(C(F)F)c1)=O N(C(=NCC(F)F)NCc1ccnn1C1CCCCC1)CC1(C(C(C)C)O)CC1 c1(C(N(C2CN(C(C3CC3CN(C)C)=O)C2)C)=O)cc2ncccc2s1 n1(CC)cnc2nc(N3CCC(c4nccs4)C3)nc(NCC(C)CO)c12 C(=O)(CC(C)(O)C(F)(F)F)N1CC(C)(C)C(NC(=O)Cc2ccco2)CC1 C(c1ccc(C)o1)=CC(=O)NC(C(=O)NC(C(=O)OCCC)C)c1ccoc1 c1(C(=O)NC2C(CNC(c3ccc(CO)c(F)c3)=O)C2)ncnc(O)c1Cl Cc1[nH]nc(C(=O)NCC2CC(NC(c3ccc(CN(C)C)o3)=O)CC2O)c1F N1(C(C2(COC)C=CCC2)=O)CCOC(CN(C)C(C2CC=CC(O)C2)=O)C1 C1(C(N2C(CO)CC(C)(C)C2)=O)CC12CCN(CC(O)CO)CC2 c1(C(N)=O)cc(C(=O)NCc2nocc2C(=O)NCCCC2CCCC2)n[nH]1 n1(CC(N2CCOCC(NC(c3nc(CC)[nH]n3)=O)C2)=O)c(C)cc(O)cc1=O C1(NC(C2CCC(=O)NC2)=O)CCCCCC1C(=O)NCCN1CCCC(O)C1 C1(NC(C(C)SC)=O)CCN(C(=O)CCn2c(C)ccc2C)C1(C)C C(=O)(CC1=CCN(C(=O)C(C)(CC)CO)CC1)N(CCCC=C)CC c1(-c2nnc(NC(C(F)=C(C)C)=O)s2)ccc(F)cc1 c1(C(N(C)CCOCCNC(=O)CC2CCOC2)=O)cc(Cl)ns1 CCC(CC(=O)N1CCC(C(=O)N2CC(O)CO2)C(C)(C)C1)C(C)(C)C S(=O)(=O)(c1cccc(=NCCC(C)CCCC(C)C)[nH]1)NC1(C=C)CCC1 c1(C(CC)C)nccc(=NCC2CCCN(C(=O)CCN3CCCS3(=O)=O)C2)[nH]1 c1(C(=O)NCC=CCNC(c2c(C(=O)OC)coc2)=O)cc(Cl)cnc1O C1(N(C(COCCCC(C)C)=O)C)CC2CC1N(C(c1cc(Cl)ns1)=O)C2 C1(CNC(c2cc(C)c(C)nc2)=O)CC2(CO1)CC(F)(F)C2 N1(C(CCCC)=O)CCN(CCCNC(=O)CC2CCN(CCN(C)C)CC2)CC1 C12(CNC(Cn3ccc(C)n3)=O)CC(CNC(=O)CC3CC=CC3)(CO1)C2 C1(CNC(C(C=CC)O)=O)CCN(C(c2nc(C)c(C)s2)=O)C1(C)C C12(C(=O)NCCC(C)C)CCN(C(=O)C(C(C)C)c3ccc(Cl)cc3)CC1C2 c1(OC)cc(F)c(F)cc1CN1CCC(O)(C(=O)Nc2ccc(C)c(F)c2)C1 n1(CC)nnc(C(=O)NC2CC(O)C2CC(=O)NCC(CC)n2cccn2)c1C Cc1cc(N)ccc1C(N1CC=CC1Cn1cc(CCOC(C)C)nn1)=O C1(C(=O)NCC(F)Cl)CCCCCCN1C(=O)Cc1cnsc1 C=CC(O)C(C)(C)C(=O)N1CC2OCC(C(=O)N(CCO)CCO)C2C1 C1(NC(c2cnc(C)s2)=O)CCC(C)N(Cc2ccc(C(F)(F)F)cn2)C1 C1(CNC(c2c(OC)c[nH]n2)=O)CCN(C(=O)CCCCCNC(N)=O)C(C)C1 c1(C(=O)NC2CCN(C(=O)CCOC3CCCC3)C2)ccc(C2=CCCC2)cc1 C1(c2cn(CCCC(=O)OCC)nn2)CC(OC)CN1C(=O)C=C(C)I N1(C(CCOCCOC)=O)CCCC(N(CCF)C(C2CCCO2)=O)C1 N1(C(C=Cc2nc(C)sc2)=O)CCC2(CCCC2NC(=O)Cc2occc2C)C1 c1(CC(N2C(C)CC(CNC(C3(CC=C)CC3)=O)C2)=O)c(C)nn(C)c1C C(=O)(CS(=O)(=O)CCO)NC1CCC(N(C(CSCCC)=O)C)CC1 C1(C(=O)NC2(C(=O)NCCC3CC(OC)C3)CCC2)CCCC(CSC)C1 S(=O)(=O)(c1cccc(=NC2CC(CC(N)=O)C2)[nH]1)NCC1COCC(C)(C)O1 n1(CC)nc(C(=O)NC2CCN(C(=O)C(CCOC)OC)CC2O)ccc1=O C=C(F)CN=c1[nH]c(=NCCc2ccncc2F)c2cccc(F)c2[nH]1 N1(C(=O)Cn2cc(Cl)cn2)CCC2C(CCN2C(c2cn3cccnc3n2)=O)C1 c1(C(N2CC3C(NC(=O)Cc4cncs4)(C3)C2)=O)cccc2ncccc12 N1(C(C(CCC)OCC)=O)CCN(C(=O)CCN2CCOCC2)C(CF)C1 CC(C)CC(CNC=O)CC(=O)NC1CN(C(C2CC3CC3C2)=O)CC12CC2 c1(OC)ccc(C(=O)NC2COCC2CNC(=O)CCSC2CCCC2)cc1N C1(NC(c2c(C)n(C)nn2)=O)(CNC(c2cnc(N)c(Cl)c2)=O)CCCCC1C N1(C(c2onc(CC)c2C)=O)CC(CNC(=O)CCc2cnc(C)o2)CCC1C C1(F)(COC)CCC(CNC(=O)C(=O)NC2(CC3CCC3)CC2)C1 CC1CCc2[nH]c(=NCc3cn[nH]c3)nc(N3CC4C5CCC(CC5)C4C3)c2C1 N1(C(c2cc(C(=O)OC)no2)=O)CCC(O)(C(C)NC(C2CCSCC2)=O)C1 CCC(C)C(C(=O)N1CCC(CNC(=O)CCC(C)(C)c2ccccc2)C1)OC c1(OC)ccc(C(=O)NCCN(C(=O)C(Cl)=CCl)Cc2ccc(Cl)nc2)cc1O Cc1cc(C(N2CCCC2CC(N2C3CCC2CC3)=O)=O)cc(C)c1C N1(C(CCSCCCC)=O)CCC2C(CCCN2C(=O)CCN2CCCC2)C1 c1(OC)nccnc1C(=O)NC1CCC(CNC(C2CC(=O)C2C(C)(C)C)=O)C1 C(=O)(CC(COC)NC(=O)C(COC(C)=O)OC)NCCCCC C(=O)(CCCN(C)C(C1(OC)CC1)=O)N(C(CC)CO)C c1(CNC(=O)Nc2cc(-c3cccc(OC)c3)on2)cc(OC)nc(Cl)c1 CCC(C)C(C(C(=O)NC1CCCCC1)NC(C)=O)N(C)C(C1CCOCC1)C C1(C)(OC)CCCN(C(=O)C(CNC(c2ncccc2O)=O)CC(C)C)CC1 CS(=O)c1cccc(C(N2CCSCC2CCNC(C2CCCCS2)=O)=O)c1 C(CCN(C)C(c1oc(C(C)C)nc1C)=O)(C(C)(C)C)NC(C(CCSC)O)=O N1(C(Cc2cn(C(C)C)nc2)=O)CCC2(CC1)CC2NC(c1cnc(O)s1)=O c1(C(=O)NCC(CC)N(C(=O)CCCCOC)C)cncc(Cl)c1 c1(OC)ccccc1-c1cnc(C(=O)NC(CSC)C(=O)O)s1 c1(C(=O)NC(N2CC(C34CC(C3)C4)CC23CCC3)=O)cnc2[nH]ccnc1-2 C=C1CC(C(=O)NC(C)CCNC(C2CC(=C3CCC3)C2)=O)(COC)C1 c1(C(=O)NC2CCCN(C(c3n[nH]cc3Cl)=O)CC2)ccc(Cl)c(Cl)c1O N1(C(c2nn[nH]n2)CC)CCC(COC(F)F)CC1 N1(C(C(COCC)C)=O)CCC(O)CC1C(=O)NOCc1ccc(O)cc1 S(=O)(=O)(c1ccc2c(c1)CCCNC2)N1CC(OC)C(C(=O)O)CC1 N1(C(c2ccc(C(C)C)cc2)=O)CCC2(C(=O)N3CC(O)CO3)CC2C1 S(=O)(=O)(c1ccc(CCC(=O)OCC(C2CCCC2)C)cc1)NC C1(C(N(C2CCN(CCC(=C)C)CC2)C)=O)CCCC(=O)N1C C1(C(C)NC(=O)CCOC2CC2)CCCCN1C(c1[nH]ccc1C1CC1)=O c1(C2(CNC(N(c3cccc(C(C)C)n3)C)=O)CC2)ccc2c(c1)OC(F)(F)O2 N1(CC(=O)NC2CN(C(C(c3cccc(F)c3)C)=O)C3C2C3)CCCCCC1=O N1(C(CCOc2c(C)cccc2)=O)CC(CO)C2(C1)CN(C(=O)CSC(F)F)C2 c1(CC)cnc2ccccc2c1C(N1CCC(O)(C(C)CNC(C)=O)C1)=O CC(C)CC(CNC(=O)C(C)Oc1ccccc1F)NC(=O)CN(C)CCO N1(C(CC(CNC(C2C3(CC3)C23CC3)=O)OC)=O)CC2CCC1C(O)C2O C1(CNC(Cc2cn(C)nn2)=O)CC12CCN(C(c1sccc1C1CC1)=O)CC2 CC1CCC(C)(C(=O)NC2CCCCC2n2cc(C3CC3)nn2)CC1 C(=O)(C1CCCc2ncccc21)NCC(CC=C)NC(=O)CCC(=C)Cl CCC(F)(F)C(=O)NCCC1(NC(c2cccc(=O)o2)=O)CCC1 C12(CNC(c3c(F)ccc(C)c3)=O)CN(C(=O)Cc3ccnn3C)CC1CCO2 c1(C(=O)NCC(CNC(=O)C=C(Cl)Cl)C(F)(F)F)cc2ccccn2n1 Cc1sc(C(=O)NCC(C)NC(=O)C(C)Oc2ccc(F)cc2)cc1Br n1(CC)ncc(C)c1C(=O)NC(C)CCCCNC(C1CN(C(C)C)CCO1)=O CCC(CC(=O)NCc1ncoc1CCNC(c1cn(C)c(SC)n1)=O)C1CC1 C1(CC)CCCCCCN1C(=O)C(CC(C)C)NC(c1cnnc(O)c1)=O C1(NC(=O)C(C2CCC(F)(F)C2)O)C=CS(=O)(=O)C1 c1(C(C)C)ccc(F)c(C(=O)NCCC(C)N(C(=O)CCC2CC2(Cl)Cl)C)c1 c1(C(N(CC(=O)NCC(C)(CO)CO)CC2CC2)=O)ccc2nccn2c1 c1(SCCC(=O)NC2C(NC(CN3CCC(C)CC3)=O)CC2)ccc(F)c(F)c1 Cn1cc(C(N2CC3CC3(NC(c3scnc3C(F)F)=O)C2)=O)c(=O)n(C)c1=O C12(C(N3CCCC(C(=O)NC(CC=C)CC)C3)=O)CC(C)(CCO1)C2 c1(OC)nn(C)cc1CNC(=O)C(Cc1ccoc1)NC(=O)C(C)CSC C1(C(N2C(C)CCC2)=O)CC12CN(Cc1cnccc1Cl)C2 C1(CC#C)(C(=O)NC2COCC2SC)CCN(C(c2cncs2)=O)C1 C1(CC(=O)NCC(C)(CO)NC(C(N2CCOCC2=O)C)=O)CC(=O)NC1=O c1(NC(C2CCCN(C(CC)=O)CC2)=O)cccc2cnccc12 c1(CC)cc(C)ccc1C(=O)NC1CCCC1CNC(=O)CC1CC(O)C1(C)C N1(C(COc2cn(C)nc2)=O)CC2C(CCNC(=O)CC3CCOC3)C2C1 Cc1ccnn1C(C)C(=O)NCC1(C(=O)NC2(CF)CCC2)CCCO1 C1(C(=O)NCCC(=C)CNC(=O)C(F)CC(C)C)CC2(CCCCC2)S1(=O)=O CCCCCCC(F)C(=O)NC1COCCN(C(C2CCCCNC2=O)=O)C1 NC(=O)CC(C(=O)N1CCC1C1CCCC1)NC(C1CCC2(CCC2)C1)=O CN1CCC2(CCN(C(C3CCC(CNC(C4(C)CC5CC5C4)=O)O3)=O)C2)C1 N1(CCC(N2CC(OCCNC(c3cnc(Cl)[nH]3)=O)C2)=O)CCCS1(=O)=O CC#CCCCC(=O)NC1CCC(NC(c2cn(C3CCOCC3)cn2)=O)CC1 c1(SCC(=O)NCC(C2CCC2)NC(C(F)=CC)=O)nnc(S)s1 C1(CN(C)Cc2ccc(N3CCCC3)o2)CCc2cc(I)ccc2O1 CCC(C(=O)N1CCC1CNC(=O)C(=O)N(C)C)N1CCCC1=O CC(C)(CO)C(C1CC1)NC(c1conc1CNC(C1(F)CC=CCC1)=O)=O C1(OC)(OC)CC(C(=O)N(C)CCN(C(C)C)CC(c2ccsc2Br)=O)C1 Cc1cc(C(=O)NC2CCCN(C(C3(C)CC4(CC4)C3)=O)C2)ccc1O Cc1cccc(CC(=O)NCCNC(c2n[nH]c3c2COC3)=O)c1F Cn1nc(C(=O)NC2CC2NC(C2(C(F)(F)F)CC2)=O)cc1F c1(C(N(C(CN(C(c2c(C)cc[nH]2)=O)C)C)C)=O)ccc(C(N)=O)nc1 C(=O)(C#CC1CCCC1)NC(C(C)(C)NC(Cn1nc(C)c(C)c1C)=O)C CCC(C)C(CC(=O)NCCC(C)C(C)C)NC(C1(CC)CCC1)=O c1(OC)c(CN2CCC(F)(C(=O)Nc3cc(C(N)=O)nn3C)C2)cccc1Cl c1(N(CCOC)CCNC(C2CCCC3CC23)=O)nc(C)ncc1C Cc1ccc(Br)c(C(=O)NC2CCN(C(C3CC=CCC3)=O)CC2(C)C)c1F c1(C(=O)NCCCN(C(=O)CNC(C)=O)CC)sccc1C(F)F N1(C(CC(C=C)C)=O)CC(C)(C)OCC1CNC(c1nn(C)cc1SC)=O c1(CC(N2CCCC(F)(CNC(CCC3(C)CC3)=O)C2)=O)cccc([N+](=O)[O-])c1 C1(NC(c2cc(C)no2)=O)CCC(C)N(C(=O)CCOc2ccc(F)cc2Cl)C1 CC1(C(=O)NCCOCCNC(c2ccn(C(F)(F)F)n2)=O)C=CCC1 C(C(=O)NC12CC(C)(C1)C2)(C(C)(C)C)NC(CC1(C)CC1)=O c1(OC)ccc2[nH]c(=NCC3CC3)nc(N3CCN(c4nc(C)cs4)CC3)c2c1 c1(C(=O)NCCN(C(C(C)SCCCC)=O)C(C)C)oc2ccc(Cl)cc2c1C C1(NC(c2cccc(CC)n2)=O)CCCN(C(=O)CCc2ccc[nH]2)C1C C(=O)(CCS(C)=O)N(C1CCN(C(=O)C=Cc2cn(C)nn2)C1)CCC C(=O)(C1=C(C#N)CCC1)NC(CC(C)C)C(=O)N1CCC1C1CCOCC1 c1(CCC(=O)NCCNC(C2(C)C(C)(C)C2)=O)ccc2c(c1)OCO2 N1(C(C(C)OCCOC)=O)CC(O)(CCNC(=O)C(C(=O)OC)NC(C)=O)C1 C1(C(N2C(CN(C(c3n(C=C)ncc3)=O)C)CC(F)C2)=O)CN2CCN1CC2C C(=O)(NNc1ccc(F)nn1)N1C(c2c(C)nn(C)c2C)CCC1 N1(c2n(CCCOC)c(C)nn2)CC2CCC(COC=CC(C)(C)[N+](=O)[O-])(C2)C1 c1(CN2CCC(CCCCCNC(C(C)=C3CC3)=O)CC2)ccc(O)cc1F c1(C(=O)NC2(C)CN(C(C(C)CF)=O)C2)ccc(N2CCC(C)C2)cc1 CC(c1cccs1)=CC(=O)NCCC1CSCCN1C(C1CCC(F)CC1)=O Cc1cccc(C(=O)NCC2CN(C)CCN2C(C2CC3CCC2C3)=O)c1N N1(C(=O)CN2CCOC2=O)CCC(CO)(NC(=O)COC2CC2)CC1 N1(C(c2c(NC)scn2)=O)CCC(NC(=O)C=CC(F)(F)F)C(C)(C)C1 c1(C2(C)CC2)cc(C(=O)NC2CCCC2CNC(=O)Cc2cc[nH]n2)no1 N1(C(CCn2c(C)ncc2)=O)CCN(C(c2csc(C)c2C)=O)C(CC(F)F)C1 c1(C(=O)NC(C(C(C)C)NC(=O)C2=NNC(=O)CC2)C)cnc2ncccc2c1 C#CCCC(C(=O)NCC(C1CCC1)OC)NC(C1CCCC(=O)C1)=O C1(CCNC(c2c(CC)ocn2)=O)CCCCN1C(=O)CCNC(=O)C(C)(C)C N(C1c2ccccc2CC1NC(c1csc(S)n1)=O)C(C1C(C(C)O)C1)=O c1(NC(C2CC(F)CN2C(c2cc[nH]c2)=O)=O)cc(Br)cc2cc[nH]c12 C=CC1(CC(=O)NC2CN(C(=O)C(C3CCC3)C3CCC3)CC2C)CCCCC1 N1(C(CCC)=O)CCN(C(=O)C2CC2)C(=O)C1.C1(CC(=O)O)CC2CCC1C2 C#CC1(NC(C2(NC(=O)C(C)n3cccn3)CC2C)=O)CC(F)(F)C1 CC1CN(C(c2cccc(CO)c2)=O)CCN1C(C1CC2CCC2C1)=O c1(C(=O)NCC23C(CN(C(C4C(CCC)C4)=O)C2)C3)cccc2cc(O)ccc12 Cc1cccc(CN(C(=O)C(C)C)Cc2cccs2)c1 Cc1ccc(N(C(=O)C(C)CN(C(=O)C(C)n2cncn2)C)C)cc1C C1(NC(=O)CC2(CO)CC2)CCCCC12CCN(c1ncnc3c1COC3)C2 [N-]=[N+]=NC(CCC(N)=O)C(=O)N1CC2CC1C2NC(C1CCc2nn[nH]c2C1)=O C1(C(N2CCCC(C3N(C(C)=O)CCC3)C2)=O)CCCC(C)(C)O1 N1(C(c2cc(I)ccc2Br)=O)CCCC2C1CCN2C(c1ccc(O)cc1F)=O c1(-n2c(C)nnc2)ccc(C(=O)NC(C)CCNC(=O)C(C)n2cncn2)cc1 Cc1cnc(Cl)cc1NC(=O)NC1CCC1C N1(CC)CC(O)CC1Cn1nc(C)cc1C.n12cc(nn1)C2 n1(CCNC(c2n(CC)nnn2)c2cnc(C(F)F)s2)nc2ccccn2c1=O Cc1ncc2n1CC(C(N1CCCC(N(C(=O)CP(C)(C)=O)C)C1)=O)CC2 Cc1cc(I)c(F)cc1NC(C1CCCC(NCc2cccc(CO)n2)C1)=O c1(CNC(=O)C(O)CNC(=O)COC2CC2)ccc(O)c(F)c1 C=CC(CC)CC(=O)NCC1CCCCN(C(=O)CN2CCN(C)CC2)C1 C1(NC(C(C)OCC)=O)CCC(C)(CNC(c2sc(F)cc2Cl)=O)CC1 N1(C2CCN(CN3C(=O)c4c([nH]c(=N)s4)C3)C2)CCC23CCCCC2(C1)C3(F)F c1(-c2c(C(N(C)CCNC(C3CC3F)=O)=O)cccc2)cccc(C#N)c1 C1(C(=O)NCc2ccnc(F)c2)C2CC(O)C(C2)N1C(C1CCCSC1)=O C1(C(=O)NC(C2(O)CN(C(c3cc(C(F)F)cs3)=O)C2)C)CN(CP(C)(C)=O)C1 C(=O)(CC(C(C)C)C(C)C)N1CC(NC(c2c(C)nc(COCC)s2)=O)C1 c1(CC)cnc(N2CCC(C)C2CNC(=O)C(C)Cc2c(C)n[nH]c2C)nc1 C=CCC(CCCCC)C(=O)N1CC2CC(NC(c3ccoc3)=O)C1C2 c1(CC(N2CCC(N(C(=O)CCN3CCOC3=O)C)C2)=O)ccc(F)nc1 N1(C(C2(CNC(C(C3CC3)SC)=O)CCCC2)=O)CCCCCC1C CC1CN(C(C2(CF)CC2)=O)CC(CNC(=O)CC2CCCC3CC23)O1 N1(C(C(=CC2CCCC2)C)=O)C2CC1CN(C(=O)C(C)n1cccn1)C2 C1(C(N2CC(CNC(C3CC4C(C3)C4(F)F)=O)C2)=O)Cc2ccncc2C1 c1(CC(N2CCCC(Cc3c(C)cccc3)C2)=O)c(Cl)ccc(O)c1Cl c1(CC(C(=O)NCCC(=C)CNC(c2cnc(C)[nH]2)=O)C)c(C)nn(C)c1C C12(CNC(CC3(C)N(C(COC4(C)CCC4)=O)CC3)=O)CCC(CC1O)C2 N1(CC(=O)Nc2cn(C)c(=O)cc2)Cc2n[nH]cc2CC1C(=O)O C1(C(N(CC)Cc2ccccc2I)=O)C=CCNCC1 c1(C(N(C(C)CNC(=O)CCP(C)(C)=O)C)=O)sc2cc(F)ccc2c1Cl N1(C(c2ccc(F)c3c2CNC3)=O)CCS(=O)(=O)CC12CNC2 CC1=NN(C)C(=O)C1CC(=O)NCCCCNC(c1sc(C(C)(C)C)nc1C)=O c1(C(=O)NC2CC(C)N(C(=O)Cc3cc(O)nc(O)n3)C2)cn2c(n1)CCCN2 C(=O)(C1=C(C#N)CCC1)NC(C1CCOC1)CNC(CCCc1c(C)ccs1)=O c1(OCCCC(=O)NCCNC(C2CCCCS2)=O)ccc(F)cc1F CCC(CC)C(F)C(=O)N1CC=CCC1C(=O)NOCC(C)C CN1CCC(CC(=O)NCCOCCCN(C(=O)CO)C)C1=O C12(NC(CCNC(=O)OC)=O)CCN(C(c3ccc(CC4CC4)s3)=O)CC1C2 c1(NCC2CCN(C(c3cc(OC)c(O)c(Cl)c3)=O)C2)ncnc2cnccc12 c1(CC)ncncc1C(=O)NCCC(C)(C)NC(=O)Cc1cc(C)on1 CCCC(CNC(c1c[nH]c2cnccc12)=O)C(=O)NOCC(C)CC c1(C(c2onc(C(C(CC)CC)C)n2)(C)C)cc(F)ccc1F CCCC(CC)CC(=O)NCC(O)CNc1nccc(OCCC)n1 C1(C(=O)NCC2CC(O)(CNC(=O)CN3C(=O)CCC3=O)C2)CC2(CCC2)CO1 C1(C(=O)NC(c2cccc(C)n2)C)CC2(CC2)CN1C(=O)Cc1csc(C)c1 C#CCC(O)C(=O)NCCn1cc(CNC(=O)C(C#N)CC)nn1 c1(C(N(CCCNC(C2CC(C)OCC2)=O)C)=O)cccc(Cl)c1[N+](=O)[O-] CC1CN(C(=O)CCn2ccnn2)CC(C)N1C(C1CC2(CCC2O)C1)=O CC1CN(C(=O)COc2cccnc2)CCC1N(C)C(c1coc2c1COC2)=O c1(C(N(CC)CC2CCCN2C(=O)Cc2cc[nH]n2)=O)csc2ccc(F)cc12 C1(NC(C=Cc2c(C)n[nH]c2)=O)CN(C(C2CC(=O)N(C)C2)=O)CC12CC2 c1(C(=O)NC2CC(N(C(COCCSC)=O)C)C2)ccc(C(C)(C)C)nc1 C(=O)(CCCCCC)NC(C(=O)NC(C#CCC)(C)C)CCOCCOC C(=O)(N=c1cc2n([nH]1)CCCC2)C1CCN(C(C2(CN(C)C)CC2)=O)CC1(C)C N1(C(C(=O)NC(c2cc(F)cc(F)c2)C)=O)CC2CCC1C(CO)C2 N1(CCN(CC(N)=O)C)CCCC(NC(=O)CCC2CC2)C1 c1(C(=O)NC(CCC)CNC(=O)C(C)CCOC)nc(C)ccc1F N1(C(CCCCOC)=O)CCC2(CCC2)C(CNC(=O)C(O)CC2CCCC2)C1 C(C1=NOC2CN(C(c3cccc(N)c3F)=O)CC12)NC(c1n[nH]c(C)c1Cl)=O C1(C(=O)NC(C)C(=O)NO)CC2(CCC2)CN1C(=O)CCCCC1CC1 c1(NC2(CNS(CC)(=O)=O)CCOC2)[nH]nc(OC(C2CC(C)(C)C2)=O)c1Cl c1(C(=O)NCCCCCNC(C2C(CCC)CCC2)=O)ccnc2c1nnn2C S(=O)(=O)(c1cccc(=NC(CO)C2CCOC2)[nH]1)NC(C)(C)CS(C)(=O)=O c1(OC)cnncc1C(N1CCCC(C(C)C(=O)NCCc2scnc2C)C1)=O C(=O)(CC(C)CC(F)(F)F)NC1CN(C(C2(CC(=O)OC)CC2)=O)CC1N=[N+]=[N-] CON=CC(=O)NC(C)(C)CN(C(=O)Cc1cncn1C)C CCC1=C(C(=O)N2CCC(C(=O)NCCN=[N+]=[N-])C2C(C)C)CCCO1 N1(CC(=O)NCC(C)NC(=O)CCN2CCC(F)C2)CCCCCCC1=O CC1=CCC(C)(C(N2CCCC(CO)(NC(C3CCCS3)=O)C2)=O)CC1 c1(C(=O)NCCC(=O)N(CCOCC=C)C)ncc(N)cc1C N1(C(C(C)c2ccsn2)=O)CCCN(C(=O)CCn2cccn2)CC1C C1(C(=O)NCCCN2CC=CC2)CCCN(C(=O)CCCF)C1 C(=O)(C(CC(C)C)ONC(C1CCS(=O)(=O)C1)=O)NC c1(C(=O)NCCN(C(CC(CC)C2CCC2)=O)C(C)C)coc2c1CCCC2 c1(C(=O)NC2CCN(C(CC3CCC(=O)NC3=O)=O)C2)cc2cccc(Cl)c2[nH]1 c1(C(N(CCCNC(CCCOCCOCC)=O)C)=O)cc(CC)ccc1Cl C1(C(=O)NCCCCCN(C(CN(C(C)=O)C)=O)C)C2CCC1(c1ccco1)C2 C1(C(=O)NC(C#C)(CO)CO)CN(C(c2ccccc2O)=O)CC1C1CC1 n1(CCCSC)nnnc1C(C1CCCO1)(C)NCc1ccn(C2CC2)n1 C1(CCNC(c2cc(C(C)C)nn2C)=O)CC(F)(F)CN1C(C1CC1(Cl)Cl)=O N1(C(c2ccc(CC)o2)=O)C2CCC1CN(C(c1cc(C3CC3)nn1CC)=O)C2 CCCCCCCC(C(=O)NC1CCOCC1)N(C1(c2ccc(O)cc2)CC1)C C(=O)(C(F)CC(CC)CC)N(C1CCC(NC(CNC(CC)=O)=O)CC1)C c1(C(=O)NCCC2(NC(c3cnc(C)[nH]3)=O)CCC2)[nH]nc([N+](=O)[O-])c1Cl C12(CNC(=O)CN3CCCC3=O)CC(CN1C(=O)Cc1csnn1)C2 C1(NC(=O)Cn2cccn2)Cc2ccccc2N(C(=O)C(F)C2=CCCCC2)C1 c1(CC(=O)NC2C(CC)CN(C(=O)CCC3CC3)CC2)cccc(S(C)(=O)=O)c1 CC1CN(C)CC1NC(C1OCCC1CNC(c1ccn(C)n1)=O)=O C1(C(N(C2CCCCC2)CCNC(C=CC=CCC)=O)=O)CCn2nccc2C1 c1(C(N2CC(O)CC(NC(C(C)=C3CCC3)=O)C2)=O)cc(C)c2nc(C)nn2c1 N1(C(CCC(C)C)=O)CCc2nc(O)cc(C(=O)NCC(C)C3CC3)c2C1 n1(CCN(CC(C)C)C(c2cn(CC(CC)O)nn2)=O)ncc2ccccc12 c1(CC)cc(C(N2CCCC2CN(C(C2CCCCS2)=O)CC)=O)c(C)nn1 c1(C(=O)NCC2CCC(NC(c3c(C)coc3)=O)C2)ncnc(O)c1F c1(C(N2CCC(CN(C(c3cc(COC)sc3)=O)C)C2)=O)ccn2c1CCCC2 c1(C(N2CC(OC)C(NC(=O)CN3CCC3C)C2)=O)cnn2c1CCC2 C(C(C)(C)COC)(c1n(C(C(=O)OC)C)nnn1)NC1CCS(=O)(=O)C1 NS(=O)(=O)c1cccc(S(=O)(=O)NC(c2c(I)ccc(Cl)c2Cl)=O)c1 C1(C(N(C(CNC(C(CC)N(CC)CC)=O)C)CC)=O)CC2(CCOCC2)CO1 N1(C(C2(CCOC)CCC2)=O)CCC(C2CCN(C(=O)CC3CCCC3)CC2)C1 c1(C(=O)NCCC(CNC(C(CC#C)C2CC2)=O)O)csc2ccc(OC)cc12 N1(C(c2c(C)nc(CC)o2)=O)CC2CC1CCN2C(=O)C(C)CC c1(C(=O)NCC(C(C)C)(C)NC(c2cnco2)=O)n[nH]c2c1CCC(C)(C)C2 c1(CNC2CC(C(=O)OC)C2)cccc2cccnc12 CN=c1[nH]c(=NCC(=O)Nc2cccc(F)c2)[nH]c(=NC(C)c2nncs2)[nH]1 C1(C(N2C(C3(C(=O)NC4CC(C)OCC4)CC3)CCC2)=O)CCCCC(=O)C1 C(=O)(C(C)(C)C(F)(F)F)NC(CN1CCN(C(C=C(C)Cl)=O)CC1)C C1(C)(CSC)C2Cc3ccccc3C12.C1CCOC(=O)N1.COC C1(CNC(c2nc(CC)sc2)=O)C(OC)C(OC)CN1C(=O)CCn1cccn1 C(CC(N)C(C)(C)C)N(C)Cc1c(N(C)C)ccnc1 Cc1cc(C(F)(F)F)n2ncc(C(=O)OCC(=O)N3CCC3)c2n1 n1(CCCOCC)c(N2CC(OCC)C(F)C2)nnc1-c1ccc(Cl)s1 C1(C(N2CCCC(NC(=O)C=Cc3cc[nH]n3)CC2)=O)CCc2cncn2C1 c1(NC(C2C=CC(NC(c3cc(C)c(F)nc3)=O)C2)=O)cccc(C#N)c1Cl C(CN=C(NCCc1ccco1)NCCN1CCCC1)c1ccc(C)nc1 CC1CC(C(=O)NCC2(C)CCN(C(=O)C(F)(F)C3(O)CCC3)C2)=NO1 Cc1ccc2sc(N3CCOC(C)(CNC(=O)C=Cc4cn(C)nn4)C3)nc2c1 Cc1cn2c(n1)CN(C(c1coc(CNC(c3n[nH]c(C)c3C)=O)c1)=O)CC2 Cc1cc(C(N2CCCC(C(=O)N(C)Cc3nncn3C)CC2)=O)c[nH]c1=N C#CCCCCC(=O)N1C(C(=O)NCCC2CC3C=CC2C3)CC1C C1(CNC(CCCC=C)=O)CN(C(=O)Cc2ccc(Cl)cn2)CC1(F)CO Cc1ncc(C(N2CCCCC2C2CCCN(C(c3ccno3)=O)C2)=O)n1C C12CC(C)CN(C1)C2=O.c1(C)cccnc1.c1(CN(OC)CC2CC2)cnc[nH]1 C1(O)(C(C)NC(c2cn(C)nn2)=O)CCN(c2nnc(C#N)s2)CC1 Cc1ncc(C(=O)NC(c2cc(Cl)ccc2Cl)c2nn[nH]n2)cc1C#N c1(NC(c2n(CC)ncn2)C)nc(=NCC2C3COCC23)[nH]c2c(C)nn(C)c12 N1(C(c2c(C)c(=O)cc[nH]2)=O)CCC(C2CC2)(CNC(c2ccccn2)=O)C1 C1(NC(C2N=C(C)SC2)=O)CCN(C(c2cc(C)ccc2O)=O)C1(C)C N1(C(C2C(NC(c3ccc(Cl)cc3)=O)C2)=O)Cc2cc(Br)cnc2C1 C=CC1(C(=O)NC2C=CCN(C(=O)Cc3cccc(NC(C)=O)c3)C2)CCCC1 C1(C(=O)NCCNC(=O)Cc2csc(C(F)(F)F)n2)CC2(CC2)CO1.c1cnco1 C(=O)(CC(C)(C)CC(F)(F)F)N1CCCC(C)(CNC(C(C)OCCC=C)=O)C1 n1(CC(=O)NCCC2CCN(C(CC(=C)Br)=O)C(C)C2)ccc(=O)n(C)c1=O c1(OCC)ccc(NC(c2cnn(CC)c2)c2nnnn2C2CCOCC2)cn1 c1(C(N(CC(CNC(C(COC)COC)=O)O)C)=O)cc(Cl)ccc1Cl C1(NC(c2ccc(COC)o2)=O)CC12CCN(C(=O)C(C)N(CC(F)(F)F)C)C2 C1(C(=O)NC2CN(C(COCCOC)=O)C2)CC(C(=O)O)C12CCC2 C12(C(=O)Nc3cn(CCC)nc3)CCCC1N(C(=O)CC1COCC(C)O1)CC2 CCC(C#N)C(=O)N(C(C(=O)N(C)CCOC(C)C)C1CC1)C C1(CNC(C2C(C)(C)NC(=O)C2)=O)N(c2ncc3c(n2)COC3)CCCC1(C)C C12(NC(c3coc(Br)c3)=O)CC3CCC(C1C2)N3C(c1cc(CF)on1)=O N1(C(CC#N)=O)CC2CCC2(CNC(c2cccnc2C(F)(F)F)=O)C1 C1(C(N(CCCCCCC)C)=O)CNC(=O)CN1C(=O)C(C)NC(=O)CC C1(CNC(C(C)CN(C(=O)C(C2CC2)N(C)C)C)=O)CC2CCC1CC2 c1(NC(C2CN(C(c3cc[nH]c3)=O)CCS2)=O)c(F)cc([N+](=O)[O-])cc1Br C1(O)CN(C(C2CC(=C3CCC3)C2)=O)CC1C(=O)NOCCCO Cc1ccc2c(c1)SC(C(=O)NCC1CC1NC(=O)CS(=O)(=O)CC(C)C)C2 N1(C(C2CC(C)(CC)C2)=O)CCC(C)C(CNC(C2(OC)CC2)=O)C1 c1(N(C)Cc2ccc(OC)cc2)ncnc2c1ncn2CCc1nc(Br)sc1C c1(C(=O)OC)nnc2ccccc2c1N1CC(CNC(=O)CC(C)CC(C)C)C1 CC(C(=O)NCC1(c2ccccc2)CC(NC(c2cccc[n+]2[O-])=O)C1)C(F)F S(=O)(=O)(c1ccc(CC(N2CC3CCC(C(=O)OC(C)(C)C)C3C2)=O)cc1)NC c1(OC)nc(C(=O)NC(CNC(=O)C=CCN(C)C)C2CC2)cc2ccccc12 C(=O)(CS(=O)CC)N(CCC(=O)NC(C#C)CCC)CCCO C(C(CCC)=C1CC1)NC(CCN(CCCCC)C1CC1)=O C1(CNC(c2c(C)n(C)cn2)=O)CC2(CC2)CN1C(C1CN(C)CCO1)=O c1(CC)nscc1NC(=O)CCOCCCNC(C1CC1C)=O C(=O)(C1CCCc2sccc21)N1C(CN(c2ccnc(C(F)(F)F)n2)C)CCC1 Cn1nc(C(=O)NC2CCOCC2NC(c2cnc(C3CC3)s2)=O)cc1C1CC1 N1(C(C(C)OC)=O)CC2CCN(C(c3cc(I)ccc3C)=O)C2C1 CC(C)(C)CCC(=O)N1CC(CNC(=O)Cc2cncc(Br)c2)CC(O)C1 C1(NC(Cc2nc(CC)sc2)=O)CCC(NC(=O)C(C)C2CCC2)CC1 C12(C(=O)NC(CC(CC)C)C)CC(CN(C(c3nccnc3N)=O)C1)C2 C(CCC1CCC1)(C(=O)N(c1ccncc1)CC)NC(CCC)=O c1(C(=O)NCC2OCC(CNC(=O)Cn3nnc(=O)[nH]3)C2)cc(F)cc(Cl)c1 S(=O)(=O)(CCCS(=O)(=O)C(F)(F)F)NC(c1cccc(CCC)c1)=O N1(C(CC2CC(=C)C2)=O)CCCC(NC(=O)CC2CC2(C)C)C1CC c1(C(N2C(CNC(=O)C=Cc3cc[nH]n3)COCC2)=O)ccc(F)c2occc12 Cc1cc(C)n2ncc(C(=O)NC3(CNC(=O)CCC4CCCOC4)CC3)c2n1 CS(=O)(=O)CC(C(C)(C)C)CCN1CCNS1(=O)=O.c1(CN)nnnn1C1CC1 Cc1scnc1C(=O)NCC(C)(C)CN(C(=O)C(C)OCCC(C)C)C N1(CCCOc2ccccc2)CCCC(C(F)F)C1.c12noc(n1)C2 c1(C(N2CCC(NC(c3cc(C)c(Cl)s3)=O)C2C(C)C)=O)cc2c(ccn2C)[nH]1 N1(C(CCC(C)C)=O)CC23CCCC2(C1)CN(C(c1ccc(Cl)c(O)c1N)=O)C3 C1(C(N(C(C)C)CCNC(c2ccnn2CC(F)F)=O)=O)CCC2(CCC2)C1 C1(C(=O)OC)CCOC12CCN(C(c1cc(Cl)cc([N+](=O)[O-])c1N)=O)CC2 C(CCC)(C(=O)N1CCCC1CN(C(=O)CC1CCCO1)C)=CCC C(C(O)C(=O)NC(C)CNC(c1ncoc1C1CCCO1)=O)=CCCC C(C(O)C(=O)NCC(O)CNC(=O)C=C1CC1)=CC(C)C c1(CCNC(c2c(C)nn(C)c2C#N)=O)cn2cccc(C)c2n1 S(=O)(=O)(c1ccsc1C(N1CCC(NC(C2(O)CC(F)(F)C2)=O)C1)=O)NC C#CCCCCCC(=O)NC(CC)C(=O)NOCCOC C1(C(=O)NC(C#C)C(C)C)(CNC(=O)CC=C(Cl)Cl)CC2(CC2)C1 C1(NC(C(C)C(F)F)=O)CCN(C(=O)C(c2ccc(Cl)nc2)(F)F)CC1O c1(C(N(CCNC(c2c(C)ncn2C)=O)CC)=O)ccc2cn(C)nc2c1 c1(-n2ccc(NC(N3CCC(OCc4ccc(F)cn4)C3)=O)n2)ccccc1F N1(C(C(C)=C2CCCC2)=O)CCC(NC(=O)CCc2cn[nH]c2)C(CO)C1 N1(CC(=O)N(C(=O)CC(C)C(F)F)CC)CC(C(c2ccccc2)=O)C(C)(C)C1 C1(C(N(CCC(=O)NC2CN(C(=O)OC)C2)C)=O)CCCC1C C1(NC(C2(C)C=CCC2)=O)CC=C(C(=O)NCCc2nnc(O)o2)C1 c1(C(N(CCN(C(C(CCSC)NC=O)=O)C)C)=O)n[nH]c2c1CN(C)CC2 CC(CCC(=O)NCC=CC1CC1)NC(C1CC2(CCC2)C1)=O Cc1ccc(CNC(C2CC2C(C)NC(=O)C2=CCCC2C)=O)cc1O c1(OC(C)C)ccc(-c2noc(CS(C)(=N)=O)n2)cc1 CC1(C(=O)NCC(O)CNC(C2(CF)CC2(F)F)=O)CCCO1 N#Cc1cc(F)c(C(=O)NC2COCC2NC(=O)CC2CC2(Cl)Cl)c(F)c1 c1(C(=O)NCC2CN(C(C=CC(=O)OCC)=O)C2)cc(C2CC2)no1 Cc1cccc(C)c1C(=O)NCC1CC(CNC(=O)Cc2cnsc2)CO1 N1(C(CCOC)=O)CCC(C2(NC(C3CC(C(F)F)C3)=O)CCC2)CC1 c1(C(=O)NC(c2cccc([N+](=O)[O-])c2)CSC)c(O)c(Cl)cc(Cl)c1Cl N1(C(C(C)(C)SC)=O)CCC(CN(C)C(c2sccc2F)=O)CC1 C(=O)(CC(C)(C)C#N)N1C(C)CC(NC(COCCCC(C)C)=O)C1 c1(C(=O)NC2CCN(C(c3c(Cl)cc(C)c(C)c3)=O)C2)ccc2c(c1O)CCC2 N1(C(C2(SC)CC2)=O)CC(O)(CN(C)C(C2CCN2S(C)(=O)=O)=O)C1 C(=O)(CCCCN(C)C)NCC(COC)NC(=O)C(COC)OC C(=O)(N=c1[nH]nc(C(=O)OC)s1)Oc1ccccc1CN(C)CC N1(C(c2c(O)ccc(N)c2)=O)CC(NC(=O)C(F)n2cccn2)C2CCCCC12 c1(C(=O)NC(CN(C(C=CC=CCC)=O)CC)C)cnc(O)c2cccnc12 c1(C(N(C2CCN(C(=O)OC(C)(C)C)C2)CCO)=O)cc2n(n1)CCCO2 N(C1CCc2ccccc21)C(C12CN(C(C3(C#C)CC(=O)C3)=O)C(C1)CO2)=O C12(CNC(CNC(CC)=O)=O)CC1CN(C(=O)C(C(C)C)n1ccnc1)C2 CC1CCCCC1(C)NC(=O)C=CC1CCN(C(=O)CC2(C)OCCO2)CC1 S(=O)(=O)(c1cc(Br)c(Br)s1)N1CCN(C(c2c(OC)nc(Br)cc2)=O)CC1C n1(CC)cc(C(N2CC3CC(C2)C3NC(C2CC2OC(C)(C)C)=O)=O)ccc1=O C=CC(C)(C)CC(=O)N1CCC(C)(NC(c2cnc(SC)s2)=O)C1 N1(C(c2nnn(C)n2)=O)CCN(C(c2sccc2F)=O)CC1c1cccnc1 C(=O)(CCCCC#N)NC(CC)(C)CNC(=O)CNc1ccc(C(N)=O)cc1 c1(C(c2nnnn2CCCCC2CC2)NCC2(CO)CC2)cnc(C(C)(F)F)s1.OC C(C)(C(=O)NC1CCCC1C(=O)N(C)Cc1ccoc1)(C(C)C)OC C(=O)(C1CC(=O)c2ccccc21)NCC1(NC(C(C)C(F)F)=O)CCC1 CS(=O)(=O)C1CCCN(C(C23CC(C(=O)NCc4cncnc4)(C2)C3)=O)C1 n1(CC#C)cccc1C(=O)N(CCC(=O)NCC1CCC(=O)O1)CC1CC1 c1(CC(N2C(C)(CNC(CCC(C)O)=O)CCC2)=O)ccc(O)c(Cl)c1 c1(C(=O)NCC(C)N(C(=O)Cn2cccc2)C)cnc2ccsc2c1 C1(CC(=O)NCCSCC(=O)Nc2cc(F)ccc2O)CCCCC12CC2 c1(C(=O)NC(C2CCN(C(C3CCC(F)C3)=O)C2)C)cc(C(F)F)[nH]n1 C1(O)(CNC(C2CC23CC3)=O)CCCN(C(c2cscc2Br)=O)C1 C1(CCCC)CN(C(=O)C(F)(F)C(C)O)CCN1C(c1cocn1)=O c1(C(=O)NC(c2ccc(C)cc2)CNC(=O)C2=CCC2)c(N)ccc(F)c1F C(N=c1[nH]c2c(c(=NCCCC3CCOC3)[nH]1)SCC2)c1c(C)cc(C)nc1 C1(C)(C(=O)NCC2(OC)CCN(C(=O)C=C3CCN(C)CC3)C2)CC2(CCC2)C1 c1(C(N(CCNC(C(CC)NC(c2ccco2)=O)=O)C)=O)cc(Br)c(C)o1 N1(C(c2cc(OC)cc(Cl)c2)=O)CCN(C(C2CCCN2N=O)=O)CC(CO)C1 C1(c2nc(-c3c(C)oc(Cc4cc(C(F)(F)F)n[nH]4)c3)on2)CCS(=O)(=O)C(C)C1 Cc1cc(CC(=O)NCCC2COCCN2C(=O)CCN(C)C)n(C)n1 c1(C(N2CC(OCCNC(c3ccncn3)=O)C2)=O)cc2cccnc2s1 c1(C(N2C(CC(=O)NCCCN(OC)C)CC2)=O)cnc(C)nc1C CC1(C)CC(C(=O)N2CCCC2CNC(c2nc(Cl)ccc2F)=O)=NO1 C1(CCNC(C2CCCSC2)=O)CCCCN1C(C1CCCN1C1CC1)=O C1(C(=O)Nc2cccc(Cl)c2)(CC)CCCN(C(c2ccnnc2O)=O)C1 C1(CC(=O)NC(CCOC)CNC(=O)CCCC(CCC)OC)CCCC(F)(F)C1 c1(C(=O)NC(CCCC)CNC(c2csnc2OC)=O)ccc2oc(O)nc2c1 c1(C(=O)NC2C(NC(CC(C)SC)=O)CCC2)coc2c1COC2 c1(C(=O)NCC2(NC(C34CCN(CC3)C4)=O)CCOCC2)ccc2n[nH]cc2c1 N1(C(CC(C)c2cnn(C)c2)=O)CCC(CNC(C2(CCO)CC2)=O)C12CCC2 C(=O)(C#CC1(C)COC1)N(CCCNC(c1c(C2CC2)ccc(C)c1)=O)C(C)C C1(NC(C2C(C=C)OCC2)=O)CCN(C(c2oncc2CC)=O)C12CCC2 c1(C2C(C(=O)NCCCCNC(c3ccnnc3O)=O)CC2)ccc(F)cc1F c1(OC)ccc(S(C)(=O)=O)cc1C(N1CCC(NC(C2COC(=O)C2)=O)C1C)=O N1(C(CP(C)(C)=O)=O)CC(CNC(C2CCC3(CCC3)C2)=O)CC1(C)C C1(CNC(C(CSC)O)=O)CC2(CCN(C(c3cc(C)cc(Cl)c3N)=O)CC2)C1 C12(C(N3CC4CC(NC(C(C)(C)CF)=O)C4C3)=O)C3C(=O)C4C5CC(C14)C2C35 c1(OCCSCc2nnc(C(C)C)s2)cc(Br)cc(F)c1F Cc1nscc1CC(=O)NCCNC(=O)CCc1cncs1 CCCCCCCC(=O)N1CCN(Cc2ccc(Br)s2)CC1C(F)(F)F C1(C)(C(=O)NCC(C)N(C(C=Cc2cncc(C)c2)=O)C)CC2CCC(C1)S2 C(=O)(C(C)(C)Cc1ccccc1)NCC1N(C(C2C(=C)CC2)=O)CC1 c1(CC)cc(C)ccc1C(=O)N(CCNC(=O)Cc1ccc(C(C)C)cc1)CC c1(C(N2CCC(C#N)(NC(C3CC=CCC3)=O)C2)=O)cc(F)c(Cl)cc1Cl Cc1cncnc1C(N1CCCC(CCNC(=O)CCc2csc(=N)[nH]2)C1)=O N1(C(C2C(C)(C)CCCC2)=O)CCN(C(c2ccc3cnsc3c2)=O)CC(O)C1 c1(CC)ccc(C(=O)NCCC2CN(C(=O)Cc3nc[nH]n3)C2)cc1Cl c1(OCC)ccc(CC(=O)NCCC2CSCCN2C(C2CC(C#N)C2)=O)nc1 C1(OC)CCn2cc(C(=O)N(C(C)CN(C(=O)C(F)=C3CCCC3)C)C)nc2C1 N1(CCNC(c2n(CC=C)ccc2)=O)CCC(NC(=O)COCC(=O)NC)CC1 C1(NC(c2cn(CC)nc2C)=O)CC2CN(C(=O)C=Cc3ccnn3C)CC12 c1(CC(N2CCOCC(C)(CO)C2)=O)noc2ccc(Br)cc12 C(=O)(C1=C(C)OCC1)NC(CN(C(C1COCC(=O)N1C(C)C)=O)CC)C N1(C(c2c(C)cncc2)=O)CCCN(C(c2ccccc2S(C)=O)=O)CC1C N1(CC(C)C)CCC(C(=O)NC2(CNC(C3CCN(CC(C)C)C3)=O)CC2)C1 C1(CC(=O)NC2(C)CC(NC(=O)CNC(C3CCCC3)=O)C2)CCS(=O)(=O)C1 N1(C(CC(CC)C)=O)CC2CCCC2(NC(=O)C(CO)N(C)C)C1 Cc1ncnc(C(=O)NC(C)(CNC(=O)C(C)(C)C2CCCO2)C(C)C)c1C c1(C(N2CC(NC(c3ccc(C=C)cc3)=O)C(F)C2)=O)c(F)ccc2ccoc12 c1(C(=O)NCCCC(C)NC(CCC=C(C)C)=O)cc(C)c(C)cc1N N1(C(CC2(C(=O)OC)CC2)=O)CCN(CC2CNC(=O)C2)C(c2ccccc2)C1 C1(C#N)(C(=O)NC(C)CN(C(=O)Cc2cnccn2)C)CC1(C)C C1(CN(C(C=C(CC)CC)=O)C)CN(C(c2oc(C(C)C)nc2C)=O)CC12CC2 c1(CC(=O)OC)cnc[nH]c1=NCCCCCCNC(=O)C1=C(Cl)CC1 N1(C(C(n2cc(CN3CCCCC3)nn2)C)=O)CC2(CC(O)CNC2=O)C1 c1(C(N2CCC(NC(CCOCC(C)C)=O)C(F)C2)=O)cn(C)c(=O)n(C)c1=O c1(NC(C2C(NC(c3cc(OC)cc(Br)c3)=O)C2)=O)cc(Cl)c(Br)cc1[N+](=O)[O-] c1(CC(=O)NCC2(CCNC(CC(C)F)=O)CC2)cc(Br)ccc1Br C(C(=O)NCC1CCC(C(=O)NCCN(CC(C)O)C)O1)(C(C)C)SC Cc1ccc2c(c1)ncn2CC(=O)NC(C)CN(C)C(c1ccc(N)cc1O)=O c1(C(=O)NCCCC(C)=O)cccc(-c2sc(C)nc2C)c1 Cc1cccc(C)c1OCC(=O)NC1CCOCC1NC(C1(C)CCOCC1)=O c1(C(N2CC(C)N(C(=O)C(CO)N(C)C)CC2)=O)cc2cccnc2cc1F N1(C(C(CC#C)NC(=O)CC2(O)CCCOC2)=O)CCC(O)(C#C)C1 Clc1ccc(C2(CNC(C3CCCOCC3)c3nnnn3C3COC3)CC2)cc1 CON1CCC(C(N2CCC(N(C(=O)CC3CC(F)C3)C)CC2)=O)CC1 c1(C(=O)NC(CC)CN(C)C(C2CC=CCC2)=O)nccc(OC)c1F N1(C(c2nc(C)oc2)=O)CC(NC(c2cc(Cl)c(Cl)s2)=O)C(O)C1 O=C1CN(Cc2c(F)ccc(CN3CCC3)c2)C(=O)C2(CCC23CCCC3)N1 N1(C(c2cc(NC(C)=O)ncc2)=O)CC2CCCC2(NC(c2cnsc2)=O)C1 N1(C(=O)CC(C(F)F)c2ccc(F)cc2)CCOc2c(Br)cncc21 c1(OCC(=O)NC2CCC2CNC(C2CC(n3cnnc3)C2)=O)cncc(Cl)n1 CCCCC(CNC(=O)C(CC)Oc1cccc(Cl)c1)NC(C1(N(C)C)CC1)=O c1(CN(C(C(N2CCC(C)CC2)C(C)C)=O)C)c[nH]c2ncccc12 c1(C(N(C(C)CNC(=O)C(C)OCC(F)(F)F)CC)=O)ccc(OC)c(O)c1 N1(C(CCNC(CC(C)C)=O)=O)CCOC(C2CN(C(c3nnc(O)s3)=O)C2)C1 C(=O)(N1CC=CCO1)NCc1n(CCC)ccc1 c1(C(=O)NC(C2(NC(C3NC(=O)CC3C)=O)CC2)C)ccc(C#CC2CC2)cc1 c1(C(N(CCCNC(C2CC(=C)C2)=O)C2CC2)=O)ccc(SC)c([N+](=O)[O-])c1 N1(C(c2c(C(C)C)n[nH]c2)=O)CC(NC(=O)C(O)C2CCC2)CC2(CCC2)C1 C(=O)(CCCC(F)(F)F)N1C(CN(C(C(CC=CCC)C)=O)C)CCC1 Cc1cc(CNC(C2(CF)CCN(C(=O)CNC(=O)CN(C)C)C2)=O)ccc1F c1(CNC2C(C(=O)NCc3ccnc(Cl)c3)CCC2)cccc(C(F)(F)F)c1Cl c1(C(N2CCC(NC(c3c(NC)cnnc3)=O)C(C)C2)=O)cc(F)c(C)cc1F CCC(CC)CC(=O)NC(C)CN1CCN(C(=O)CCc2cnccn2)CC1 C1(NC(c2scc(COC)c2)=O)CCC(C)(NC(C23CC4CC2C3C4)=O)CC1 N=c1nc(N2CCc3c(F)cccc3C2)[nH]c(=NC2CNC(=O)C2)[nH]1 c1(C(=O)NC(CC)CNC(=O)C(C)N2CCC2)cc2ccccc2nc1O NC(=O)C1=NOC(CNC(C2CCN(C(=O)C=Cc3ccsc3)CC2)=O)C1 c1(C(=O)NC(CC)CN(C)C(C2(OC)CCOC2)=O)c(C)cnn1C c1(C(=O)NCC(CC)NC(=O)C(F)(F)c2cccnc2)ccnc2ncccc12 CC1(C(N2CCCC(C(N)=O)C2)=O)CCN(C(=O)CC23CCC(CC2)C3)CC1 Cc1nn2cc(C(N3CCC(N(C(=O)Cn4cncn4)C)C3)=O)nc2s1 C1(C(=O)NC2(OC)CCCCC2)CN(C(=O)NCC(C)(C)OCCO)CC1(C)C CC1CN(C(=O)C2CC2)CC(C)N(C(=O)C=CSc2nc[nH]n2)C1 N1(C(CC(C(=O)OC)C)=O)CCC(C)(C)C(NC(c2cccnc2O)=O)C1 c1(C(N2CC(NC(c3ccc(C)c(C)c3)=O)C(O)C2)=O)cc([N+](=O)[O-])ccc1C c1(C(N2CCCCC(CO)C2)C(=O)NCCCOC)cc(Cl)c(C)cc1Br C(=O)(C1CSc2ccccc21)NCCC1(CNC(C2(C)CCCNC2=O)=O)CC1 Cc1noc(C2(NC(c3nc(CC(=O)OCC(C#N)C4CC4)cs3)=O)CC2)n1 C(=O)(C(C)C(F)(F)F)N(CCOCCC(=O)NCCN(CCC)CC)C C(c1ccc(F)cc1)=C(C)C(=O)NC1(CNC(c2coc(C(F)F)n2)=O)CCC1 C1(CNC(c2csc(O)n2)=O)CC2(CCN(C(c3cscc3C(F)F)=O)CC2)C1 c1(OCC#C)ncccc1C(=O)NCC1(NC(=O)CC2NC(=O)NC2=O)CCC1 C1(C(CNC(=O)Cc2cnoc2)NC(CSCCOC)=O)CCCCC1 c1(C(=O)NC(C)(CNC(c2cc(C(F)F)[nH]n2)=O)CO)c[nH]c2cccc(F)c12 c1(C(c2n(CCOCC)nnn2)NC(C)Cc2ccsc2)ncc(Cl)cc1Cl CCC(CC)CC(F)C(=O)N1CCC(O)(n2cc(CN(C)C3CC3)nn2)CC1 C=CCC(C)(C)CC(=O)NC12CC(NC(=O)Cn3ccc4ccccc34)(C1)C2 c1(C(=O)NC2CC3(CC(NC(=O)CCCC4CC4)C3)C2)ccn2ncccc12 N1(C(C2(CC#C)CCC2)=O)CCC(CCCCNC(C2CCC(=O)N2)=O)CC1 C1(N(CC(C)C)C(c2cnco2)=O)CCN(C(C2CCC(O)CC2)=O)CC1 C(=O)(C(C(CC)CC)N(C)C)N1CC(C=C)(CC(N2CCOCC2CO)=O)C1 c1(OC)ccc(SC(C)=O)c(NC(=O)C(N2CCC(CO)(CO)C2)C2CCC2)c1 C1(NC(C2CN3CCN2CC3)=O)C2CC1CN(C(C1CC=CCC1)=O)C2 N1(C(c2onc(C)n2)=O)CCC2(CCCN(C(=O)CCC(C)N(C)C)C2)C1 c1(C(=O)NCC(C)=CC(=O)NCC2CCCC2C2CC2)nc(C)ccc1C C1(CNC(=O)Cn2cnc(Br)c2)CC(F)CN1C(c1cccc(F)c1)=O C1(NC(C2(NC(c3c(CC)c[nH]n3)=O)CC2(C)C)=O)CCCC(C(N)=O)C1 C(=O)(CCC1=CCCCC1)N1CCC(NC(c2c(=O)ccn(C)c2)=O)C12CC2 C1(CCNC(c2ccoc2)=O)COCCN1C(=O)C1=CCSC1 N1(C(C2CCN(CC)CC2)=O)CCC(C2(NC(C3CCC4CC34)=O)CC2)C1 c1(C(N(CC(CC)NC(=O)C=CC2CC2)CC)=O)cc(C)n(C(C)C)c1 N1(CC(C)C)CCCN(C(C(=O)NC2CC(F)(F)C2)C(C)C2CC2)CC1 C12(NC(C=CCOC)=O)CC(C)(C1)OC21CN(C(c2nn(C)cc2SC)=O)C1 C1(C(N2C(C)(CNC(c3cn(C)nc3C(F)F)=O)CCC2)=O)Cc2nccn2C1 c1(CN(C)CC2(c3cnn(C)c3)CCCO2)cccc(C(=O)O)c1 C(=O)(C(=O)N=S(C)(C)=O)NC(CCCC)CNC(C1CCCC1O)=O N1(CCn2cc(CNC(C)=O)nn2)CCCN(C(=O)C(C)c2ccsc2)CC1 C(C(C(=O)NCC1CC(NC(=O)CC2CCC(C(F)(F)F)O2)C1)OC)OC Cc1ccc(-c2nc(CCSC3CCC3)n(CCCCO)n2)cc1Br C1(NC(C)=O)CCC(C)N(C(c2cn(-c3noc(C(F)(F)F)n3)cn2)=O)C1 Cc1sc(C(=O)NCCCCC(C)NC(=O)C=CBr)cc1Br Nc1cc(C(=O)NC(CNC(c2cnn(C3CC3)c2)=O)C2CCC2)ccc1Br c1(CNC(=O)Nc2c(OCC)nccc2)cccc(C)c1F Cc1nccn1CC(N1CCC1C(=O)NC1CC(n2ccnn2)C1)=O C1(CC=C)(NC(=O)C(F)(F)c2ccccc2)CCN(C(=O)CC(=O)N(C)C)C1 CC1CC(NC(c2nc(Cl)c(Cl)s2)=O)CN1C(=O)Cc1cccnc1 CC(C)CC(O)C(=O)NC1(CCCNC(=O)C=CC(=O)OC(C)(C)C)CC1 CC1(C)C(C(=O)NCC2(CN(C(=O)CCc3csnn3)C3CC3)CC2)C1C(F)F Cc1ccc(NC(c2sccc2NCc2ccc(O)c(Cl)c2)=O)c(C#N)c1 CC1(C)COCCC1NC(=NCCc1cccnc1O)NCc1ccccc1 C(=O)(C(C)(C)C(=O)NS(=O)(=O)CC(C1CCCCC1)OC)OCC CC(C)CC(C)(CNC(C1(C)C(C)(C)C1(C)C)=O)NC(C1CCCOCC1)=O C1(C(=O)NCC2C(NC(CC(CC)CC)=O)C2)CC(=O)NC2CCCCC12 N1(C(C2(C)C=CCCC2)=O)CCCC(CCNC(=O)Cc2cnoc2)CC1 CP(C)(=O)CN1CC(C(=O)NC2CCCC2CNC(c2cncc(O)c2)=O)C1 CP(C)(=O)C(O)C(=O)NCC1(O)CCN(C(c2ccc(C(F)F)s2)=O)CC1 C(=O)(CC1OCc2ccccc21)N(C(C)CNC(c1ncn2ccccc12)=O)C Cc1cccc(C(=O)N(C)CCN(C(c2ncc[nH]2)=O)C(C)C)c1[N+](=O)[O-] C(c1ccc(F)c(F)c1)=C(C)C(=O)NC(C)CN(C(=O)CC1CC1(Cl)Cl)C N1(C(C(=O)NCCCCO)=O)CCCC1C(=O)NCCCc1ccccc1 CCCC(CC)CCC(=O)NCC1CCCN1C(c1cccnc1OC(F)F)=O CN1CC(F)CC1C(=O)NC1CCC(C(=O)NC2(c3ncc[nH]3)CC2)CC1 CC#CCCCC(=O)N1CCC(NC(=O)C2CC2)C1C N1(C(CSCCC)=O)CCC(CN(C(=O)CCCc2nncn2C)CC)CC1 C1(NC(C2CC(=C)C2)=O)CC(CNC(=O)Cc2sccc2C)C1(C)C C(=O)(CC(C)(O)C(F)(F)F)NCC(C)NC(c1cccc2nc(C(F)F)[nH]c12)=O c1(C(=O)NC2CCCC(NC(CCC3CCC(=O)N3)=O)C2)cc(O)ccc1Cl n1(CC(=O)NCC(C2CCC2)NC(=O)CCn2cccc2)cc(Br)cn1 Cc1cncc(C(=O)NC(C2CC(NC(c3cnn(C)c3)=O)C2)C)n1 N1(C(Cc2cnc(C)[nH]2)=O)CCN(C(CNC(=O)C2=CCCC2)C(F)F)CC1 N1(C(C(C)S)=O)CCC(O)C(C(=O)NC2CNC(=O)C2(C)C)C1 c1(C(N2C(CC)C(C(=O)N(CC(F)(F)CO)C)CC2)=O)cccc2[nH]ncc12 C(c1cc2ccccc2o1)=CC(=O)NCC1CC(NC(C(C)N(C)C)=O)CC1O C(CCC)(C(O)C(=O)N1CCC(CO)C(C)(C)C1)NC(C(C)OCCCC)=O N1(COCC)N=C(C(=O)N2CC3CC3(CF)C2)CCC1=O.c1(C(=O)N)nnccc1C N1(C(c2cc(C)[nH]c2)=O)CCCC(C2CC2NC(c2cc3ncccc3s2)=O)C1 C(CCCC(=O)NCCCCCCNC(C1CC1(Cl)C(=O)OC)=O)OC C1(C(=O)NCCCN(C(=O)CSc2nnnn2Cc2nccs2)C)CCNC1=O N1(C(c2[nH]cc(CC)c2)=O)CCCC12CCN(C(C1CC3CC(O)C(C1)C3)=O)C2 C1(CC)CN(C(=O)Cn2ncnn2)CCN1C(c1sc(Br)cc1F)=O c1(C(N2CC(C)C(CNC(C3(C)CCC3)=O)C2)=O)cc(O)ccc1F c1(NCC(Cn2ncc(S(C)(=O)=O)c2)O)cnc2c(Cl)cccc2n1 C1(C(=O)NC2CN(C(C(C)CCc3cccc(F)c3)=O)C2)CCc2c[nH]nc2C1 c1(OC)cc(C(F)(F)F)c(Cl)c(NC(=O)NCCS(N)(=O)=O)c1 C1(CNC(C(C)CC2CC2)=O)CCN(C(C23CC(CF)(CO2)C3)=O)CC1 c1(NC(=O)NC(CSC)CO)cnc2ccnn2c1 C(=O)(C(O)C(C(C)C)OC)N(CC)CC1CCCN(C(=O)C(F)C(F)(F)F)C1 C1(CCC)CN(C(=O)C(O)C2CCCC2)CCN1C(C1CCC2(CC1)CC2)=O C1(C(N(CC(C)NC(=O)Cc2ccccc2F)C)=O)CCn2cncc2C1 c1(C(=O)NC(C(C)C)C(C)NC(c2coc(Cl)c2)=O)cccc(C(F)(F)F)c1F C(C(C)(CC)C(N)=O)NC(C=CCN(C(CC=C=C)=O)C)=O CC(O)C(F)(F)C(=O)NC1CCC(CNC(=O)CSc2ccc(F)c(F)c2)C1 C(=O)(C(C(C)(C)C)OC)NCCN(C(c1cnc(O)c(Br)c1)=O)CC C1(CCNC(C(C)OCC(C)C)=O)CCCN(C(=O)CC2CC(F)(F)C2)C1 c1(C(N2CC(CN(C(C(CCC)(C)C)=O)C)OCC2)=O)ccc2nnc(O)n2c1 C#CCC(O)C(=O)NCCC1CCCCN1C(c1c(Cl)n[nH]c1C)=O C1(OC)CCCCCC1CNC(=NCCF)NC1CC(c2cccc(C#N)c2)C1 N1(C(CC(C)c2ccco2)=O)C(CNC(=O)CC2CCCC2)CC2COCC12 c1(C(=O)NC2(CC=C)CCCN(C(=O)CSc3nncs3)C2)ccc(C#N)cn1 C1(C(=O)NCC(C)N(C(CCc2c(C)n(C)nc2)=O)C)CCC2CCC1O2 C(=O)(C1=CCN(Cc2ccccc2)C1)NCCN(C(c1c(CCC)nco1)=O)C C1(CC)(NC(=O)Cc2c(Cl)cccc2Cl)CCCN(C(c2sncc2C)=O)C1 c1(C(=O)NC2CC2C(=O)Nc2ccon2)ccc(Oc2cccnc2)cc1 C1(COC)CN(C(=O)CSc2nncn2C)CCN1C(c1ccn(CC#N)n1)=O c1(C(N(C)CC2(O)CCN(C(CC=C)=O)C2)=O)cc(Cl)ccc1OC C1(CNC(C(=O)NC(C)C)=O)CN(C(C2(C)CCNC2=O)=O)CCC1(C)C c1(CNC(CC)C(=O)N(CCN)CCC2CCC2)cccnc1Cl c1(N(C2CCC(C)(C)CC2)C)nc2ccccc2nc1NC1CCN(C)CC1 Cc1c(F)ccc(NC(=O)C=Cc2ccc(F)c(F)c2)c1F Cc1cc(CNC(=O)CCCC2(NC(=O)C(F)OC(F)(F)F)CCC2)cnc1Cl N1(CCNC(c2ccc(O)nc2)=O)CCN(C(C23CC(O)C2C3)=O)CC1 C1(C)(C(N(C2CCN(C(C(C)C3CCC3)=O)C2)CC2CC2)=O)CCN(C)C1 C1(NC(CC=CC=C)=O)CCSC12CN(C(c1c[nH]nc1-c1cccnc1)=O)C2 C1(F)(CNC(C(C)Cc2cnco2)=O)CCN(C(c2ccc(CO)o2)=O)C1 N1(C(c2ccc(CC)[nH]2)=O)CCC(C(=O)NCc2ccncc2)C1C c1(C(c2n(CCC)nnn2)NC(C2(Cc3ccccc3)CC2)C)ccncc1Cl c1(C(=O)NC(CNC(c2cc(CC)nn2C)=O)CC)cccc(S(N)(=O)=O)c1C C1(C(=O)NCc2cn(CC(=O)N(CC(=O)N(CC)CC)C)nn2)CC(=O)N(C)C1 N1(C(c2c(C)sc(O)n2)=O)CC2CC1CN2C(=O)CC1CCCNC(=O)C1 c1(C(N(C2C3CN(C(=O)CC(C)(C)C4CC4)CC23)C)=O)ccc([N+](=O)[O-])o1 c1(NC(C(=O)NCc2cn(C(C(=O)OC)(C)C)nn2)=O)ccn2ncccc12 Cc1cccc(CC(N2CC(OCCNC(=O)Cc3ccccc3O)C2)=O)c1Cl C12(OC(C)=O)CC(C(N3CCC(C(C)NC(=O)C=CC(C)(C)N(C)C)C3)=O)(C1)C2 C1(NC(c2cc(Cl)c(F)cc2O)=O)CN(C(=O)CC2(CO)CC2)CC1C1CC1 CS(=O)(=O)C1(C(=O)NCC=CCNC(c2cnn(C3CCCC3)c2)=O)CCCC1 O=C(NNc1ccc(F)cc1Br)c1cc2ccc(Cl)cc2nn1 c1(C(=O)NC2CCCCN(C(C(C)=C3CCC3)=O)C2)c(C)nc(C2CC2)nc1O C(CN=c1[nH]c(N2CC(CO)C(C)C2)nc2ccccc12)c1c(C)n(C)nc1 C(CO)(CO)(C(=O)O)NC(C1CCN(Cc2ccccc2)C1=O)=O C(=O)(C(C)CC(F)(F)F)N(CC(=O)NC1C(C(C)C)CCC1)C1CCC1 C#CC1(C(=O)NCc2ccccc2CN(C(=O)C(CSC)OC)C)CCCC1 c1(N2C(C(=O)Nc3c(I)ccc(C)n3)C3CCC2C3)ccn2ncc(Br)c2n1 Cc1c(C=CC(=O)N(CC(C)(C)CNC(=O)C(C2CCOCC2)O)C)cnn1C CC(O)C(F)(F)C(=O)NC1COCC1CNC(=O)Cn1cnc(=N)[nH]1 c1(C(N2CCC(C)(CCNC(C3CC3C3CC3)=O)C2)=O)ncc(N)cc1Cl n1(C(C)C)ccc(=NC(=O)C2CCC(C)CN2C(C2CC3CCC3C2)=O)[nH]1 c1(COC2(C)CCC2)ccccc1CNC(=O)NC1CCCC(=O)O1 N1(C(c2n[nH]c(C)c2Cl)=O)CC(CNC(C2CC2F)=O)OC2CCCC12 C(=O)(C1=CC2CCCC12)N1C(Cc2cn(C)nc2)CC1 C(C(C)(C)C#CC(=O)NC(CO)CCCO)NC(CCCCN(C)C)=O C1(n2cc(CCCC(C)(C)C)nn2)(CS(N2CC(OC)C2)(=O)=O)CCCOC1 Cc1ccc(SC(C)C(=O)N(C)CC2CN(C(=O)C(C)(C)C#N)CCO2)cc1 c1(COC)n[nH]c(=NC2CC(CCNC(=O)C(C)(O)C3CC3)C2)s1 N1(C(C(CN=[N+]=[N-])NC(C2C(C)(C)C2)=O)=O)CCOCC2(CCC2)C1 CCCC(CCC)C(=O)NC1CCCCC1NC(=O)CC1CCOC1=O C1(N(C(c2cc(C)nn2C)C(=O)NC2CCOC2)C)CN(C)C(C)(C)C1 c1(N(C2CCOCC2)CC(N)=O)c([N+](=O)[O-])cnc2ccc(C(C)(C)C)cc12 Cc1cc(C)n(C(C)C)n1.C1(c2nnnn2CCC2(C)CC2)(N)CSCSC1 c1(C(N2C(CC(=O)NC(c3ccccc3)C)CCC2)=O)ccccc1Cl CN=c1[nH]c(C(=O)NC(CNC(=O)C(c2cccc(Cl)c2)C)C(C)(C)C)cs1 C1(C(=O)OC(c2ccccc2Cl)C)CCc2ccccc2C1O C1(N(C(C2CC(OC)C2)=O)C)CN(C(=O)Cc2cccnc2F)CC1(C)C c1(C(N2CCC(CNC(=O)CC3NC(=O)NC3=O)CC2)=O)cnc2c(c1)COC2 N1(C(CCCCOCC)=O)CCCC(O)(CN(C)C(C2CC(C(F)F)C2)=O)C1 Cc1cccc(F)c1-c1cn(CC2C(CNC(=O)OCC)C2(F)F)nn1.C(C)(C)(C)O N1(C(C2C(OC)C2)=O)CCC(C)(CNC(c2ccccc2OCC(N)=O)=O)CC1 C(CCCCC(=O)N1CCCC1CCCNC(C1CC1C1CC1)=O)SC C(C(C)(C(=O)NCC(C1CCN(C(=O)COC2CCOC2)CC1)O)OC)OC Cc1csc(=O)n1CCC(=O)NCC(F)CNC(=O)COc1cnn(C)c1 C12(NC(C3C(=C)C3)=O)CCC(CNC(c3cn(C)c(=O)cc3OC)=O)(CC1)OC2 CCCC(O)C(=O)N1CC(NC(c2cc(-n3cccc3)ccn2)=O)C(CC)C1 N1(C(c2occ(C)c2)=O)CC2CC(C1)CN(C(C1CC1c1cccs1)=O)C2 c1(C(=O)NC2CC2NC(C2CC2(Cl)Cl)=O)cc(F)cc(Br)c1 c1(C(=O)NCC2C(NC(C3(C)SCCCS3)=O)C2)cc2occc2[nH]1 CC1(C)OCCC1C(N1CCC(OCCNC(=O)CNC(c2ccccn2)=O)C1)=O c1(CN2CCCC(NC(C3CCN(C)C3)=O)C2)ccc([N+](=O)[O-])cc1O C1(CNC(c2n[nH]cc2Cl)=O)CCCCN1C(c1coc(C2CCC2)n1)=O C1(C(N2CCN(C(CNC(C(F)=CCC)=O)C)CC2)=O)Cc2nc(C)cn2C1 N1(C(CC2C(CC)C2(F)F)=O)CCOCC1CCNC(c1ncc(F)cn1)=O Cc1ncc2c(n1)CCC(NC(=O)CSc1ccccc1O)C2 c1(C(N2CC(C)C(NC(=O)CCn3ccnc3)CC2)=O)cnn2c1CCCC2 CC(C)(C)C(CNC(c1csc(Cl)c1)=O)C(=O)N1CCC(c2cnco2)C1 N1(C(c2cc(C)c(C)o2)=O)C(C)CC2CN(C(c3cccc(C4CC4)n3)=O)CC12 c1(NC)nc(C)ccc1C(=O)NC1CC(NC(=O)CCCC2CCCC2)C(O)C1 N1(C(CC(CC)SC)=O)CCC(C)(C)CC1C(=O)NCCc1ccccn1 N1(C(c2cc(OC)ncn2)=O)CCC2CC2(NC(=O)C=Cc2ccoc2)CC1 N1(C(=O)OCC)CSCC1C(=O)NC1CC(NC(=O)C=CC2CCOC2)C1 C1(NC(=O)C=Cc2sccc2Br)CC2CC(NC(C3(O)CC3)=O)CC12 N1(C(C2(N(C)C)CCC2)=O)CCC2(C=C(C(=O)N3CC(O)CC3CO)C2)C1 C1(NC(C2C(CC)CCC2)=O)CC1C1CCCN(C(=O)C(C)C)C1 Cc1cc(Cl)c(C(N2CC3CC(NC(C4(N5CCCC5)CC4)=O)C2C3)=O)cc1N Cc1cnc(N(C)CC2CCN(C(=O)C(C3CCOCC3)C)CC2)nc1C N1(C(C(CC=C)c2ccccc2)=O)CCCC(O)(c2cn(C(C)CC)nn2)C1 C=C(Br)CC(C)(C)C(=O)N1CCC2(CC1)CC2C(=O)NCCSC Cc1[nH]nc(C(N2CC3CC(NC(C4CCOCC4)=O)CC3C2)=O)c1[N+](=O)[O-] C1(N(C(c2ccncc2)CCC)C(c2ccco2)=O)CCNCCC1C c1(OC)cc(OCc2cccc(-c3cccc(N)c3C)c2)c(N)cc1F c1(C(N(C2CCN(C(C(C3CCC3)OC)=O)C2)C)=O)nn(C)nc1Br C1(CCN(C(=O)Cc2ccoc2)C)CCCCN1C(=O)C(O)Cc1ccccc1 Cc1ncc(CC(N2CC(NC(=O)COC3CCOC3)CC(F)C2)=O)c(O)n1 C1(CCN)(NC(=O)CN2CCOCC2)CCCC1.c1(C(=O)NCCCOC)ccncc1 Cc1c(C(F)(F)F)n[nH]c1C(=O)NCC(C)CN(C(=O)CN1CCC(O)CC1)C C1(C(=O)NCC23CCC(CC2)N3C(C2CC23CCC3)=O)CC1C1CCCCC1 C1(C(N(CCC(C)NC(C2(C)CCOCC2)=O)C)=O)CCOC1(C)C c1(C(=O)NC2N(C(C(COC)C)=O)CC2)ccc(OCc2cccc(C)c2)cc1 c1(C(N2CC(CNC(c3occ(C)c3)=O)C2)=O)cnn2cc(C(N)=O)cnc12 c1(CNC(C2CCC(CNC(CSCCOC)=O)C2)=O)ncccc1Cl N1(C(CC2CN(C)C2)=O)CCC2CN(C(C3CC(=C4CCC4)C3)=O)CC2CC1 C1(C(=O)NCC(C=C)(C)C)C2CC1N(C(c1c[nH]nc1OC)=O)C2 NC1CC2(CCC(c3cn(Cc4cnc5ccc(F)cn45)nn3)CC2)C1 C(CCCCCCO)NCC(=O)NC(C1CCC(NC(=O)C(C)(C)C)C1)C CC(C(=O)NC1(C)CCN(C(=O)C2=CC3CCCC23)C1)C(C)S(C)(=O)=O C(CCC(CO)NC(=O)C(C)=C1CC1)NC(C(C)N(CC)CC)=O c1(C(=O)NCC(CN(C(=O)CCNC(N)=O)C)O)cnc2sccn12 C(C(C)(CO)NC(=O)CN(C)C1CC1)NC(CC=C(C)C)=O c1(C(C)=O)ccc(CC(=O)NCC(Cc2ccccc2)N(C(=O)C(N)=O)C)cc1 c1(CC)cc(N)ccc1C(=O)NCC1(NC(=O)C(F)=CCCF)CCCCC1C O=C(CCC(F)(F)F)Nc1nc(C2CC(F)CN2Cc2ccc([N+](=O)[O-])[nH]2)n[nH]1 C1(NC(C(CSCC)NC(=O)C(CC)N(CC)CC)=O)CC2(CNC(=O)O2)C1 C1(NC(c2c(C)cccc2Cl)c2n(CCC)nnn2)CCn2ccnc2C1 C1(CC)(NC(C2OCCC2C)=O)CN(C(=O)CNC=O)C1 C1(CNC(C2CC(=O)NC2)=O)CCC(F)(CNC(=O)Cc2cnc(C3CC3)[nH]2)C1 c1(CC(N2CC3C(NC(CC=C(C)C)=O)C(C3)C2)=O)cc(F)c(F)cc1F c1(C(N2CCC(C(N(CC=C)CCO)=O)C2CC)=O)cc(C#N)[nH]c1C N1(CCc2nc(C(=O)OC(C)(C)C)sc2)CCOC(Cc2ccccc2)C1 c1(C(=O)O)c[nH]c2cc(C(=O)N(CCC(F)=C(F)F)CCO)ccc12 N1(C(CC2C(CC)C2)=O)CCC(CF)(NC(=O)CSc2nnnn2C)C1 Cc1cccc2nc(CNC(=O)C(=O)Nc3ccc(C4CCNCC4)nc3)cn12 c1(C(N2CC(N(C)C(c3scnc3Cl)=O)C2)=O)ccc2c(c1)C(=O)CCO2 C1(NC(C(C2CC(F)(F)C2)OC)=O)CC(Nc2cncc(Cl)n2)C1(C)C C12(C(=O)NC3(CC=C)CCC3)CCCC1CCN2C(=O)Cn1cc(CO)nn1 c1(C(N2CC(NC(Cc3n(C)ncc3)=O)C2)=O)cnc2c(c1)ncn2C C=C(C)CC(C(=O)NCC1CCC(NC(=O)CCOC(C)=O)C1)OC c1(C(N2C(C)C(NC(=O)C(F)(F)c3cncs3)CC2)=O)ccc2nn[nH]c2c1 c1(C(=O)OC)cc(NCC2CCSC(C)C2)nn2c(Br)cnc12 c1(C(N2C(CC)CN(C(c3ncnn3C)=O)CC2)=O)cnc2cccc(Cl)c2c1 C(CCC(C)(C)NC(=O)CC1CCN(C(=O)CN2CCCC2C)CC1)OC c1(CCC)occc1C(=O)NCC(CO)NC(=O)Cc1cn(CC)nn1 CC1(C)C(C)(C)C1(F)C(=O)N(CCC(=O)Nc1ccc(F)c(CO)c1)CCO CC(=O)C(C)CC(C)C(=O)NCC(C)(C(C)C)NC(=O)C1=CC(C)(C)C1 CC1(C(=O)NCC2CCCC2NC(=O)CSCc2cscn2)CC1(F)F N1(C(c2n(C)nc3c2CCCC3)=O)CCCCC(N=c2cc[nH]cc2[N+](=O)[O-])C1 N1(C(=O)COC(F)(F)F)CCC2C(C1)CN2C(=O)CC1CCSCC1 CC1=C(C(=O)NCC2CCCCN(C(=O)Cc3nc(=N)[nH][nH]3)C2)C(C)(C)CCC1 N1(C(C2N(C(=O)OC(C)(C)C)C(=O)CC2)=O)CCC(O)C(F)CC1 n1(CC)nc(C(N2CC(NC(=O)CCc3nc[nH]n3)CC(O)C2)=O)ccc1=O C1(NC(C(CC)=CC)=O)(CO)CCN(C(c2cc(Br)cn2C)=O)C1 N1(C(CCCCC)=O)CCCC(C)C1CNC(C1(N2CCOCC2)CC1)=O S(=O)(=O)(c1ccc(Br)cc1NC1COc2ccccc21)N1CCCCC(CC)C1 C1(c2nc(CNC(=O)CN(C(c3ccnnc3S)=O)CCO)on2)CC2CCC1C2 N1(C(Cc2c(C)scc2)=O)CC(C(=O)NC2CCC(CO)C2)C2(CC2)C1 Cc1c(C(=O)NCC2(O)CN(C(=O)C=Cc3ccn(C)c3)C2)cnn1CC(C)C C1(C(=O)OC)CC2(C1)CC(c1nnnn1C1CCOCC1)(NC1CCS(=O)C1)C2 c1(C(N2C(CNC(c3c(NCC)cccn3)=O)CC2)=O)c(F)cc(C)cc1Cl C(=O)(CCS(=O)(=O)C(F)(F)F)N1C2C(CNC(=O)COC3CC3)(CCC2)CCC1 C1(OC)CN(C(=O)CCCNC(C)=O)CC1NC(c1cc(CC2CC2)on1)=O c1(C(=O)NC2CCC(NC(=O)CCC3CCOC3)C2)ccn2c1CCCC2 c1(C(C(N2CC(NC(=O)Cn3nccn3)C2)=O)O)cccc(F)c1 Cc1nc(O)[nH]c1C(=O)NCC1(CO)CCN(C(C2(C)CC=CCC2)=O)C1 C1(C(N2CCCC(F)C2)=O)(CC)CCN(C(=O)CCOCCCOC)CC1 C12(COC)CC(NC(c3cc(C)ncc3C)=O)(CN1C(=O)Cc1ccco1)C2 c1(C(=O)NC2CN(C(C=CC=CC)=O)CC2O)cc2cncc(Br)c2s1 CC1(CNC(c2scnc2C(F)(F)F)=O)CCN(C(=O)Cc2ncc(Cl)s2)C1 C1(NC(CSn2c(C)ncc2)=O)CN(C(=O)CCCN2CCCCC2)CC1(C)C c1(CC)cccc(CC)c1C(N1CCN(C(C2(C#N)CCCO2)=O)CC1)=O C(=O)(C(C)S(C)(=O)=O)NCC(C)(Cn1cccn1)NC(C(C)CF)=O N1(C(C2(C(N)=O)CC2)=O)CCN(C(C2C=CCCC2)=O)C(c2ccccn2)C1 c1(C(=O)NCCN(C(C(C)OC)=O)CC(C)O)cc(O)c2sccc2c1 Cc1n[nH]cc1C(=O)NC(C)C(=O)NCC(C)Cn1cccn1 C1(C(N2CCC(CN(C)C)C2)=O)CN(C(=O)CC2CCC(C)(C)O2)CCN1C c1(C(=O)NC2CCN(C(=O)C(C3CCOCC3)F)CC2F)cccn2nnnc12 Cc1ccc([N+](=O)[O-])c(C(N2CCC(NC(=O)Cc3conc3C)C(C)C2)=O)c1 CCC(C)(CNC(=O)C(c1ccco1)NC(=O)Cn1ccc(C)n1)C(N)=O c1(CC)[nH]nc(C(=O)NCCOC2CCN(C(c3cc(F)c[nH]3)=O)C2)c1Cl c1(CCC(=O)NC(C(C)NC(COCCSC)=O)CO)c(F)cccc1Cl C1(C(N2C(C(=O)OC)CC2C)=O)(CO)CCN(C(C2CN(C3COC3)C2)=O)C1 CCCCC(CC)C(=O)NC(CC)CCCC(=O)NCCCCOCC Cc1ncc(C=CC(=O)NC2CN(C(=O)CC(C)(O)C3CC3)CC2C)s1 Cc1cc([N+](=O)[O-])ccc1N1CCC(C)C(NC(C2CC(CC3CC3)C2)=O)C1 C1(CC)CN(C(c2ccsc2SC)=O)CCN1C(C1CC(O)CN1CC)=O C1(N(C(=O)COC2CC(F)(F)C2)C)CN(C(C2CCCCN2S(C)(=O)=O)=O)CC1O C(CN=c1[nH]cnc(C)c1C#N)C1CCC(NC(CC(CC)CN(C)C)=O)C1 C1(C(=O)NC2C(F)CCN(C(c3c(CC)[nH]c(=N)s3)=O)C2)CCc2nn[nH]c2C1 CCN=c1ccc(C(=O)N(C)CC2CCCN2C(c2cccnc2S)=O)c[nH]1 N1(C(CSCC(C)C)=O)CCC2CN(C(c3cc4cccn4c(O)n3)=O)CCC12 C1(CNC(c2n(C)ccn2)=O)CN(C(=O)C=C2CCOCC2)CCCO1 c1(C(=O)NCCCC2N(C(C(CC=CC)C)=O)CCCC2)ccc(OC)c(N)n1 C1(C)(COC)CCN(C(=O)C(CN(C)C)NC(c2cscn2)=O)C1 C(=O)(C1=NOC(C)(C)C1)N1CCCC(CCNC(c2ccc(SC)o2)=O)CC1 C1(C(N2CC(C)(NC(C3(CC(=O)OC)CC3)=O)C2)=O)CC12CCCCC2 CCC(CC(=O)NC(C)(CO)C(=O)NC1(C)CC(O)(CO)C1)CC(C)C C1(CNC(=O)C(O)C2CCC2)CCN(C(C2CCS(=O)(=O)C2)=O)C12CC2 CC1CCc2sc(C(=O)NC3(CF)CCN(C(C4CNC(=O)N4C)=O)C3)cc2C1 Cc1ccc(Cl)cc1C(=O)N(CC(C)CNC(C1CC1[N+](=O)[O-])=O)C C=C(C)CC(C)C(=O)NCCC1CCN(C(=O)CCc2cnn(C)c2C)C1 C1(NC(c2n(C)nnc2)=O)CCN(C(=O)CCC23CCC(CC2)C3)CC1(C)C S(=O)(=O)(c1ccc(Cl)cc1F)N1CCN(Cc2ccc(CSCC)o2)CC1C C1(CC)CN(C(C2CCN(C)CC2)=O)CCN1C(=O)CC(O)C(C)C C(=O)(CC1=CCCCC1)N1CCCC(CN(C)C(C2COCCOC2)=O)C1 N1(C(c2cc(C)ncc2)=O)CC(NC(c2csc(Br)c2)=O)CC(C)C1 C1(C)(C(=O)NC2CN(C(CNC(C(CC)C)=O)=O)CC2O)C(C)(C)C1(C)C CN1CCOC2(CN(C(C3C(CNC(=O)CSCC(F)F)C3(C)C)=O)C2)C1 c1(CN(C(N(C2CCN(C)CC2)CCO)=O)C2CC2)c(S(N)(=O)=O)cnn1C c1(CCCC)nc(C)c(C(N2CC3CC2C3NC(C2CC(OC3CC3)C2)=O)=O)s1 N1(C(CC(C=C)C)=O)CCC(C)(Cn2cc(-c3cc(C)n(CC(F)(F)F)n3)nn2)CC1 C1(CC(=O)NC2C(=C)COC2)COC2(CCC2)CN1 c1(CNC(C)C)nc(C(=O)O)cs1.C(=O)C(F)=C1CCCC1.CN1CCN1C C(C(C)(C)CC(=O)NCCNC(=O)Cc1cccc(C#N)c1)N(C)C Cc1oc(Cl)nc1C(=O)NC(C(=O)NC12COC(CN(C)C)(C1)C2)C1CCCC1 c1(CN2CC3C(C(N4CCN(CCOC)CC4)=O)(C3)C2)cc2ccccc2[nH]1 N1(C(c2c(C(C)C)c(F)cnc2)=O)CCN(C(c2ccc(Br)cc2)=O)C(C)C1C c1(CCC(=O)N(CCN(C(=O)C(C)OC2CCOC2)CC)CC)nnc(C(C)C)o1 C1(C)(CCC)CCN1C(=O)C(C)CNC(=O)C(C1CCCCC1)F c1(C(N2CC(O)(CNC(C(C)Cn3ccnc3)=O)C2)=O)noc2c1CCCCC2 N1(C(c2cn(C)nc2)=O)CC2CS(=O)(=O)CC2(CNC(C2(CCO)CC2)=O)C1 C1(NC(C(C)OCCN(C)C)=O)CC2CCC1CN2C(c1n[nH]cc1Cl)=O c1(C(N2C(CNC(c3csc(C)c3N)=O)CC(F)C2)=O)nnc2n1CCCC2 c1(C(=O)NCCC(C)(C)NC(C2CCCOC2)=O)ccc2oc(=N)[nH]c2c1 c1(CCC)cccc(C(=O)NCC2CCN(C(=O)C(C)NC(=O)NC)C2)c1 C1(C(N2CC(C)(NC(C(C)=C3CC3)=O)CC2(C)C)=O)C2C3CC4C1C1C2CC3C41 C1(N(C(C(CC)OC)=O)CC)CCCN(C(=O)Cc2scnc2-c2cccs2)C1 C1(c2nnnn2CCSC)(NC2(CC=C)CCSCC2)CCCC(CC)CC1 Cc1cnc2cc(C(=O)NC3CCC3NC(c3cc(C(F)F)ccn3)=O)ccn12 C(=O)(C1=CCCCCC1)NC1CCN(C(c2cn(C(C)(C)C)nn2)=O)CC1CO C1(NC(C(C)O)=O)CS(=O)(=O)N(C)C12CCN(C(=O)CN1CCCC1C)CC2 C1(C(N2CCC3(C2)CN(C(C2CC4CCC(C2)C4)=O)C3)=O)CN2CCCN1CC2 C(=O)(C(=O)N=S(C)(C)=O)NCCO.c1(OC)cnccc1C(N1CC(C=O)C1)=O Cc1ccn(C)c1C(N1CC(NC(c2cc(CN(C)C)no2)=O)C1)=O CC1=C(C(=O)N2CCC(C(C)NC(c3ncoc3C3CCC3)=O)C2)SCCO1 C1(OC(C)(C)C)CN(C(=O)COCCF)CCN1C(=O)C(F)C1CC1 c1(C(N2CC(CNC(CC(=C=C)C)=O)C3C2C3)=O)ccc(OC)c(F)c1F N1(C(c2cc(C)nn2C(C)(C)C)=O)CCC2CCN(C(c3ccsc3)=O)CC2C1 C1(C(=O)NCCC(C)NC(c2nc(C)oc2)=O)CCCC(CF)C1 C1(CN(C(c2c(C(C)C)nns2)=O)C)COCCN1C(C1CCCCC1)=O c1(OC(CNC(CN)=O)C)ccc(I)cc1.C1C=CC1 C12(NC(C(C)CNC(C3CCO3)=O)=O)CC3CC(CC1C3)C2 C#Cc1ccc(Cl)c(C(N2CC(NC(C3(C)CCCC3)=O)CC(O)C2)=O)c1 C1(NC(c2cc(OCC)n[nH]2)=O)CCN(C(C2CCC(C(N)=O)N2C)=O)C1C N1(C(c2cc(OC)n[nH]2)=O)CCCC(O)(CNC(C2CC3CCC2O3)=O)C1 C1(C(N2CCC(F)(CNC(c3cc(CCC)n(C)n3)=O)C2)=O)CCN(C)C(=O)C1 c1(C(=O)NC2CC(CNC(CNC(=O)OCC)=O)C2)c[nH]cc1C1CC1 CC(O)CCCCCC(=O)N(C1CC(NC(=O)C=C2CCN(C)C2)C1)C C1(C(N2CCC(N(C(=O)CCCNC(c3ccco3)=O)C)C2)=O)C(Cl)(Cl)C12CC2 c1(N2CCCC(CN(C)C(C3CCC3)=O)C2)cc(C(F)F)nc(Cl)n1 C1(CC(=O)NC2CC(CCNC(CN(C3CCC3)C)=O)C2)NC(=O)CN(C)C1=O CC1(C)CC(C(=O)NCC2(C)CC3CC3C2)CN1C(=O)Cn1cncn1 c1(NCC(CC)CC(F)(F)F)ccc(S(=O)(=O)NC2CCCCC2N(C)C)cn1 CC1(C)CC(NC(=O)CC23CC(C2)C3)CCN(C(=O)Cc2cscn2)C1 c1(C(=O)OC)c[nH]c(=NCC(C)CNC(c2snnc2C)=O)c2ccsc12 CC(F)CC(=O)N1CCC(CNC(=O)C(C)OCc2ccncc2)C1 C1(C(N2C(C)CC2C(=O)NCCc2c[nH]nc2O)=O)CC2CCC2C1 c1(C(=O)NCCC(=C)CNC(c2ccc(C)nc2)=O)ccccc1SC(F)F c1(OC)cncc(C(=O)NCC=CCSCc2ncccn2)c1 C1(N(C(C(CC)c2ccccc2)=O)C)CN(C(c2cnc(=N)[nH]c2)=O)CC1(C)C CC(C)CC(C)C(=O)N1CCCC(NC(=O)CCNC(=O)Nc2ccccc2)C1 CC(C)(CC(=O)NCc1cccc(OCCO)c1)c1cccc(Br)c1 c1(C(=O)NC2C(C)N(C(=O)Cn3cnccc3=O)CC2)cc(F)cc2ccoc12 c12cccc(n1)CN2.N1(C(C2C(C(=O)O)C2)=O)CCN(CC(F)F)CC1 N1(C(C(C)SCC)=O)CCC(CCNC(c2ncc(N)nc2C)=O)C(F)(F)C1 N1(C(Cc2c(C)scc2)=O)CC(NC(=O)C(C)CSCc2cccnc2)C(O)C1 N1(C(c2cc(C)cc(C)c2)=O)CC2CCCC(NC(=O)CC(C)P(C)(C)=O)(C2)C1 N1(C(CC2CCCN(C)C2)=O)CCC(C(=O)NC2COC(=O)C2)C12CCC2 c1(C(N2CC(C(N(C(C)C)CCF)=O)OCC2)=O)cnn(C)c(=O)c1 C(=O)(C(=O)N=c1ccn(-c2ccccn2)[nH]1)NCC1CN(S(C)(=O)=O)C1 c1(OC)ccc(C(N2CCCCC2CNC(C2(OC(C)C)CCOC2)=O)=O)nc1 CC(=O)CCCCC(=O)N1CCCCC(CCC(=O)NC(C)(C)CN(C)C)C1 N1(C(C2C(C)(C)CO2)=O)CCC(F)(CNC(c2cc(Br)ccn2)=O)C1 Cc1cnn(CC(=O)NCC2CC2CC(N2CC(CCN(C)C)C2)=O)c1 C([N+](=O)[O-])C1(OCCOCC)CC1.C1(=O)COC(=O)N1.C1CO1.CO n1(CC(=O)NC2CN(C(=O)CCC3CC3)CC3(CC3)C2)ncc2ncccc12 C1(CNC(c2c(CC)csc2)=O)CC(F)(F)CN1C(=O)CCN(C)CC N1(C(C(=O)NCC)C2CC2(Br)Br)CCN(CC(c2ccccc2)=O)CC1 C=CCC(CNC(=O)CCCc1cccs1)NC(C1CCN(C(C)=O)C1)=O C1(CNC(C(COC)C)=O)CN(C(=O)CC(C)(F)F)CC2(CCC2)O1 c1(-c2cc(NCc3c(C)cnn3C(C)C)sc2)cccc2[nH]ncc12 C1(NC(=O)C=CC2CCCO2)CS(=O)(=O)C12CCN(C(C1(CF)CCC1)=O)CC2 C1(CNC(c2cnc(C)s2)=O)CC2(CC(NC(=O)C(C)c3ccsn3)C2)C1 c1(C(=O)NCC2N(c3nnc(C)o3)CC2)ccc(NC(c2ccccc2)=O)cc1 c1(C(=O)Nc2c(C(=O)NC(C)C(F)(F)F)c(F)ccc2)cc(Br)cc(F)c1F N1(C(C2(CC=C)CC=CC2)=O)CCN(C2CCN(C(c3cncs3)=O)C2)CC1 Cc1sc2nc(C(C)NC(=O)Nc3cnn(CC(C)C)c3C)nc(O)c2c1C Cc1cccc(CC(N2CCC(CNC(=O)CN(C)S(N)(=O)=O)C(O)C2)=O)c1F N1(C(C2C(C)CCC2)=O)CCC(N2CCC(NC(c3cc(O)cs3)=O)C2)CC1 C=CC1(C(N2CCC(CNC(c3ccc(F)cc3N)=O)C2)=O)CCOCC1 C(=O)(C(CC(C)C)C(C)N(CCC(C(C)(C)C)NC(=O)OC(C)(C)C)C)OCC N1(n2cc(CNC3(C(=O)NCc4c(C)noc4)COC3)nn2)CCCC(C)C1 c1(CCC(=O)NCCN(C(C(C)C)=O)C(C)C)nc(-c2ncccn2)no1 c1(C(N2C(c3cnc(C)nc3)CCC2)=O)cc(Cl)c(C(F)F)cc1F C12(NO)CCC(C(=O)NC34CC(NC(c5ccc(F)c(CO)c5)=O)(C3)C4)(CC1)C2 C(=O)(CC1=Cc2ccccc2C1)NCC1CC(OC)CN1C(C1CCC(O)C1)=O N1(C(C(=O)OCC)=O)CC(CC(=O)Nc2cnc(C)c(OC)c2)OC2(CCC2)C1 N1(C(C(C)C(C)(F)F)=O)CCCC2(C1)CN(C(=O)CCCc1cnn[nH]1)CCO2 c1(N2CCCC(C)CC2)nc(=NC2CCC(F)(F)C2)[nH]c2c1cnn2C Cc1cc2cc(C(N3CCN(C(C4CCC(CO)CC4)=O)C4CC34)=O)ccc2[nH]1 c1(CC(=O)NCCC2CCN(C(c3cc(C)c(C)o3)=O)CC2)cn2ccsc2n1 CC(C)C(C)(CNC(c1cnn(C)n1)=O)NC(=O)C=Cc1cn(C)cn1 C(=O)(CC(C(F)(F)F)c1ccccc1)N(C1CCN(C(=O)Cc2cnsc2)C1)C CC(C)(C(=O)NCc1nocc1C(=O)NCc1cscn1)n1cccn1 c1(CC(=O)NC(CNC(C2(COC)C=CCC2)=O)(C)C2CCC2)cccnc1C N1(C(c2n(CC)cnn2)=O)CC2(CCN(C(=O)CC3CCCNC3=O)C2)C1 C(=O)(CC(C)(C)C(=O)NC(CNC(=O)Cc1nc2ncccn2n1)CC)OCC C(CC(C)C(=O)NCC1CN(C(=O)CC2(Nc3ccccc3)CC2)C2CC12)=CC Cn1ncc(C(N2CCC(CCNC(c3c[nH]nc3-c3ccc(Cl)s3)=O)C2)=O)n1 Cc1ncsc1C=CC(=O)NCC#CCNC(c1cc(Br)n(C)c1)=O C(CCN(C(=O)Cc1csc(Cl)c1)C)(C(C)(C)C)NC(C1(COC)CCOC1)=O C1(CNC(C2(C)CC2Br)=O)CCCCN(C(=O)CSC2CC2)C1 C1(C(=O)NC2C(NC(c3n(C)c(S)nc3)=O)CC2)COc2ccccc2C1 C(c1ccccc1)=CCNC(CN(CCOC)C)=O.C1(=O)C(C)=CC(C)N1 N1(C(=O)Cn2cc(Cl)cn2)CCC2(CCCN2c2cc(-c3ccoc3)ncn2)C1 N1(C(C=CC(N)=O)=O)C2CCC1C(NC(=O)CCCn1ccnc1)C2 c1(C(N(C2CC(NC(C3(C4CC4)CC3)=O)C2)C)=O)cnn(-c2ccccc2)c1N N1(C(CCN(C)CC)=O)CC2CCC(N(C)C(c3cc(C)cc(Cl)c3)=O)C2C1 c1(C(=O)NC2C3CN(C(CNC(=O)NC)=O)C2CC3)cc(F)cc(C)c1N c1(C(=O)NC23CC(NC(C(CC)N(C)C)=O)(C2)C3)cccc(OC(C)(C)C)n1 c1(CC)ncccc1C(=O)NC(C)(C)CCNC(=O)C(C)C(C)C C(=O)(C1=NOC(NC(=O)C(C2CC2)OC)C1)N(CCCN(CC)CC)C C1(CC(=O)NCC(C)NC(C2(C)CCCC2C)=O)CC2CCC1O2 Cc1ncc(NC(c2ccnc(CNCc3n[nH]cc3Cl)c2)=O)nc1C c1(C(c2nnnn2CC2(C)CCCS2)NCCOC(C)C)sc(Br)nc1Cl c1(N2C(CNc3cc(OC)c(C)cc3)CNCC2)ncnc2cc[nH]c12 c1(NCc2n(CC)nnn2)cccc(OCC#N)c1.c12cncn1C2 C1(CNC(CCCOCCC)=O)CCN(C(c2c(C)noc2CC)=O)CC1(F)F C(c1cccnc1)=CC(=O)NCC1(CC(=O)NC(CC)C(C)O)CC1 C1(CNC(CC(C)(F)F)=O)C(C2CC2)CCN1C(=O)Cc1nc(C2CC2)cs1 n1(CC)nc(C2CC2)cc1C(=O)NCC1CC(C)N(C(=O)CC2(C)CC2(Cl)Cl)C1 CC1(C(N2CCC(C)(C(F)(F)F)CC2)=O)CCCN(C(c2ccccc2I)=O)C1 C=C=CCCC(=O)N(C1CCCC1)CCCNC(=O)CNC1(c2ccccc2)CC1 C1(C(N(C(C)CNC(=O)C=CCOCC(F)(F)F)CC)=O)CCN(C)CC1 c1(N(CCC)C)ccc(C(N2CCCCC2CN(C(=O)C2=CCSC2)C)=O)cc1 N1(C(CCc2n(C)ccn2)=O)CCN(C(=O)CCC2CC(F)(F)C2)CC1 CCC(CC)C(C)N=c1cc[nH]cc1S(=O)(=O)NC1CC2(CCCCCC2)C1 N1(C(C(=Cc2ccccc2)OC)=O)CCN(C(c2cnc(C(C)C)[nH]2)=O)CC1C CC12CC(C(N)=O)(C1)C1(CCN(C(=O)OCCOC3CCCO3)CC1)O2 FC(F)C(CN=c1cc(NCC(=C2CCCC2)F)nc[nH]1)c1ccccc1 C1(NC(COC2(C)CCCC2)=O)CCN(C(C2CC23CC(O)C3)=O)C12CCCC2 C(=O)(C#CC1(C)COC1)N(C)CC1(O)CCN(C(C23CCC(C2)C3(C)C)=O)C1 Cc1cc(C(=O)O)cc(CNC(c2cc(Cl)c(Br)[nH]2)=O)c1 C#CC1(C(=O)NC2CN(C(c3cnc(S)n3C)=O)CC2SC)CCCC1 C1(CC)CC(C(=O)NCCCN(C(=O)CC2CC3CC3C2)C(C)C)CCO1 N1(C(C(CC)CO)=O)CC2CCN(C(C3CC=CCC3)=O)CCC2C1 O=c1n(Cc2nc(-c3ccc(F)cn3)no2)nc2ccccn12 c1(C(=O)NC2CC3(CC(NC(=O)CCn4cccc4)C3)C2)cc2sccc2cn1 N1(C(c2ccc(OC)cn2)=O)CC2CS(=O)(=O)CC2(NC(c2cscc2F)=O)C1 c1(C(N2CCC(C3N(C(CCC)=O)CC(C)C3)CC2)=O)ccc2c(c1)CNC2=O C1(OCCNC(C2CN(C(COCCCC)=O)C2)=O)CCCCC1n1cccc1 C12(C(N3CCC(C(C)(C)NC(CC(CC)OC)=O)C3)=O)CCC(C#N)(CC1)CC2 C#Cc1ccnc(C(=O)NCC(C)CNC(=O)Cc2cccc(C(C)C)c2)c1 CCC(CC(C)O)NC(C1(SC)CN(C(c2csc(C)n2)=O)C1)=O C(=O)(C1=C(F)CN(C(=O)CCCC(C)=O)CC1)NC(CCC)CC N1(C(CC=CCC)=O)CC(NC(=O)CCc2nc(-c3cccs3)no2)CC1(C)C c1(CNC(C2CCCN2C(=O)CC2CCNC2=O)=O)cccc(O)c1 N#Cc1c(Cl)nsc1NCC1CCCCC1NC(C1CC12CCCC2)=O C1(C)(C(N2CC(CC=C)(NC(=O)Cn3ncnn3)C2)=O)Cc2ccccc2NC1=O C=CC(C)(O)CC(=O)N1CCC(N(C)C(c2ccc(CO)cc2F)=O)CC1 c1(C(=O)NC2C(C)N(C(C3CC4CCC3CC4)=O)CC2)cncc(F)c1Cl Cc1ccc(N)cc1C(N1CCC(NC(=O)CCF)C(O)C1)=O N1(C(C2CC(C)N2C(c2cscn2)=O)=O)CCc2cnccc2C1 N1(C(C2N(C)CCC2)=O)CCC2CN(C(C3CC(C)(O)C3)=O)C2C1 c1(C(=O)NC2C(OC)CN(C(C(CC#C)O)=O)C2)ccc(OC)nc1F N1(C(C(C=C=C)C)=O)CCN(C(C2(CC)CC(C)(C)C2)=O)CC1C C1(CNC(C(c2ccccc2)OC)=O)C=CC(NC(=O)CCc2ccncc2)C1 N1(C(C(CC)=CC)=O)CCN(C(c2cc(C)c(N)cn2)=O)C2CCCCC12 c1(OC)ccc([N+](=O)[O-])cc1NC(C1COCCN1Cc1cnc(Cl)c(Cl)c1)=O C1(NC(C2CN(C(C3(F)CCOCC3)=O)CCS2)=O)CC2C(=O)NCC(=O)N2C1 Cc1cc(C(N2CCC(OCCNC(=O)C(C)C3CC3)C2)=O)c2c(c1)CCC2 C(=O)(C(C1=CCSC1(C)C)N1CCC(C(C)(C)C#N)CC1)NCC(=C)C c1(-c2ccc(OC)cc2C)cccc2[nH]c(C(=O)NC3CONC3=O)cc12 C(=O)(C(CNC(=O)Cc1cc(C)nn1C)C(C)(C)C)NC(C#C)(C)CC C(CC1=CCN(C(=O)CCc2cnco2)CC1)NC(c1cn(CC)nc1)=O C1(C(N2CC(CCNC(COCCCC)=O)OCC2)=O)CC2(C1)CC2(F)F n1(CC)cc(CC(=O)N(CCCNC(C2CC3CCC2C3)=O)C(C)C)c(C)n1 N1(C(c2cc(C)sc2C)=O)CC(=O)NC2CN(C(=O)C=Cc3cncs3)CCC12 c1(C(N2CCC(N(C(=O)C(C3CC3)SC)CC)C2)=O)cc2nc(C)cc(C)n2n1 Cc1noc(C)c1CC(=O)NCCNC1(n2cc(CC(O)C3CC3)nn2)CC1 C1(C(N(CCCNC(=O)CSc2ccc(C)cc2)CC)=O)COC2(CCC2)C1 CC(O)C(C(=O)NCCCNC(=O)CC1(C)CC(F)(F)C1)NC(=O)OC(C)(C)C N1(C(CC(C)(C)C)=O)CC(NC(C2CCNC2=O)=O)CC2(CCOCC2)C1 N1(C(COCC(C)(C)C)=O)Cc2[nH]cnc2CC1C(N)=O N1(C(C=CC)=O)CCCC1CC(N1CC(C2CC2)C1)=O.C12CC(C1)N2C N1(C(Cc2c(C)nc(C)s2)=O)CCC(NC(=O)CC2CCCO2)C(F)C1 C1(C2CCCN(C(=O)C=Cc3ccccc3)C2)(NC(COCC=C)=O)CC1 Cc1nc2cc(Cl)cc(C(=O)NCCN(C)C(C3CC(=C(F)F)C3)=O)c2[nH]1 CC1(C)CC2=C(C(=O)N1)C(c1cnccc1CN)NC(=S)N2CCC#N C12(C(=O)NCCN(C(CC3CC(=C)C3)=O)CCC)CCCCC1OCC2 c1(SC)cccc(C(N2CC3CC2CN3C(c2cc(O)n(C)n2)=O)=O)c1Cl N1(C(c2c(CC)nco2)=O)CC(O)CC1(C)C(=O)NCc1cccc(O)c1C C1(C(=O)NC2CN(C(C(CC#C)(C)C)=O)CC2(C)C)CCn2cc(C)nc2C1 C1(NC(c2ccc(N)cn2)=O)CC2CCCC(C1)N2C(C1CCCC1)=O N1(CC(=O)NCC23N(C(C(C(CC)C)C)=O)C(CC2)CC3)CCCCCCC1=O N1(CC(=O)NC(C(C)C)(C)CNC(c2cc(O)ncn2)=O)CCCCC(O)C1=O C12(C(=O)NCCC3(NC(CC(C)c4cnn(C)c4)=O)CCC3)CCC(CC1O)C2 C(=O)(CS(=O)(=O)CCOC)NCC(CC)N(C)C(c1ccc[n+]([O-])c1)=O N1(C(COCCC=C)=O)CCC(NC(c2cccc(N(C)C)c2)=O)C(C(C)C)C1 c1(C(=O)NCC2CC(C)N(C(=O)CCCC(F)F)C2)cccc2nsnc12 C1(CNC(C2(OC)CCC2)=O)CCC(C)N(C(=O)CCCC2CCCC2)C1 C1(NC(CC(C)C2CC2)=O)CC2(CCN(C(c3cncn3C3CC3)=O)CC2)C1 N1(CCC)C(=O)CCC1C(=O)NC(C)CC(C)NC(=O)C(C)C1CC1 N1(C(CCCOCC)=O)CC(NC(c2cc(C(C)(C)C)oc2C)=O)C2CC12 c1(C(N2CC(C)C(NC(=O)CC3C=CCCC3)C2)=O)c[nH]c2c(C#N)cccc12 c1(OCC(N2CCC(NC(c3nnc(C)o3)=O)C2)=O)cccc(F)n1 C1(C(=O)NCCCOCCNC(C(n2ccc(C)n2)(C)C)=O)CCC2C1C2(F)F c1(C(=O)NC2C(CNC(c3ccn(CCOC)n3)=O)CCC2)cccc(F)c1C c1(NCC(C)CNC(C2CCSCC2)=O)ccc([N+](=O)[O-])c(OC(C)(C)C)c1 C(C(C(C)C)C(C)C)N(CCOC)C(c1cc(C2CC2)n(C)c1C)=O N1(C(C(C=C)(C)CC)=O)C(CNC(=O)CN2CC3CC3C2)CC2COCC12 N1(c2ncc(C)cn2)CC2CC1CN2C(c1ccn(-c2cccc(F)c2)n1)=O c1(CC(=O)NCCCN(C(C2CCC2C(N)=O)=O)CC2CCCC2)csc(S)n1 N1(C(c2cc(SC)oc2)=O)CCCC2CN(C(c3cc(=O)cc(Cl)[nH]3)=O)CCC12 C(=O)(CCCC(F)F)N(C(C)CCNC(=O)CSC(F)(F)F)C.NC C1(CC(=O)NCCN(C(=O)Cc2sccc2C)CCC)CC(C)=NO1 C1(C(=O)NC)CCN(C(=O)CC2CC3CC3C2)C1CC(=O)OC.c12cn(nn1)C2 c1(C(=O)NCCC2(CNC(C34CCCC3C4(F)F)=O)CC2)ncnc2ccsc12 CC(CC1CCC1)N=c1[nH]c(=NCc2cc(Cl)nc(Cl)c2)[nH]c2cccc(F)c12 C1(CC(=O)NC2C(C)CC=CC2)CCN(C(=O)CSC2CC2)C1(C)C C1(N(C(=O)COC(F)F)C)CCCC(NC(C2(C#N)CCC2)=O)C1 N1(C(CCNC(C)=O)=O)CCC2(NC(=O)Cc3nnc(C)o3)CCCCCC12 C1(C)(NC(COCCCC#C)=O)CCN(C(C2(OCC)CCCCC2)=O)C1 C1(NC(C(C(C)O)C)=O)C2CC3CN(C(=O)C(O)Cc4cnc[nH]4)C1C3C2 c1(OC)ccc(CO)cc1C(=O)NC(C1CCCCN1C(C1CC(F)C1)=O)C Cn1cncc1-c1cn(C2CCN(C(=O)C(C)(O)c3ccsc3Cl)C2)nn1 c1(OC)cnccc1C(N1CCC(C)C1CNC(=O)CCc1cccnc1C)=O C(=O)(CCCN=[N+]=[N-])N(C1CC(C#N)C1)CC(=O)N(CCCC(C)(F)F)C Cc1ccc(C(C)CC(=O)NC(C)Cn2cc(-c3cc(C(=O)O)cs3)nn2)cc1 C1(C(=O)OC)CCCC1S(=O)(=O)NC1CCC(Oc2ccc(F)cc2)CC1 N(C(=NCCc1cccs1)NCc1ccnn1C)Cc1ncc(C)nc1 N1(C(=O)Cc2cc(Br)cs2)CCCC(C2CN(C(C3OCCO3)=O)C2)C1 C1(C(=O)NC2CCCC2NC(C2CCOC(=O)N2)=O)(OCC)CCOCC1 C1(NC(C(F)=CCC)=O)CCC2CCN(C(c3cc(C)n(CC)c3C)=O)C1C2 CC1(CO)CCN(C(C2(NC(c3sccc3Cl)=O)CC(F)(F)C2)=O)C1 CCC(C)C(O)C(=O)NCCCCCCN(C)C(c1ccn(C)n1)=O C(C)(CCNC(C1CC1CF)=O)NC(COCCC)=O c1(C(N(CC(C)NC(c2scnc2C(C)(C)C)=O)C)=O)ccc(F)cn1 Cc1cc(C(N2CCOC(CCCNC(=O)CC3C(C)C3(F)F)C2)=O)nc(O)c1 c1(C(N2CC(C)C(CNC(=O)C(C)SC(C)C)CC2)=O)ccn2c1CCCC2 C=C(C)CC(C(=O)N(CCOC)CC)NC(c1n[nH]c(C)c1O)=O c1(SCCNC(c2n(C(C(=O)OC)C)nnn2)=O)cccnc1Cl C1(N(C(C(C)SC)=O)C)CCN(C(c2c[nH]nc2C(F)F)=O)C1 N1(CC)CCCN(Cc2cc(Cl)cc(C)c2N)CC1C(C)C C1(C(=O)NC2CCC2)CN(C(=O)C=Cc2cocn2)C2(CCC2)C1 c1(N2CCC(CN(C)CC)CC2)cc(NC(c2ccncc2F)C)nc(C)n1 C1(CCC(=O)N(CC(F)Cl)C)CCN(C(c2ns[nH]c2=O)=O)C1 C1(CN(C(C(C)OC2CCCC2)=O)C)CCCC1C(=O)OCc1ccccc1 CCS(=O)CC(=O)NC(CCN(C(=O)C=Cc1cn[nH]c1)C)C(C)C C#Cc1ccc(F)c(NC(=O)C=CC(=O)N(C(C)CCNC(=O)CCC)C)c1 c1(CNC(CC2C(CNC(c3c(CC)ncnc3)=O)C2)=O)ccc(F)c(O)c1 N1(C(C(CC)=CC)=O)CC(CNC(=O)Cn2cc(C3CC3)nn2)C(C)(C)C1 c1(C(=O)NC(CC)CNC(c2cc(C)on2)=O)ccc(S(N)(=O)=O)s1 Nc1cc(C(=O)NC2CN(C(=O)CC3CCCC(C(F)(F)F)O3)C2)cc(O)c1Cl c1(OC(C)(C)C)ccc(OC2C3CN(C(=O)NC(=O)C(C)(CO)OC)CC32)cc1 Cc1cc(C(N2CCN(C(=O)CSc3n[nH]c(O)n3)CC2C2CC2)=O)cc(C)c1 N1(C(C2COCCN2C(=O)CCc2cnc[nH]2)=O)CCC2(CCCNC2=O)CC1 N1(C(Cc2c(C)con2)=O)CC(NC(=O)CCS(C)(=O)=O)CC12CCCOC2 c1(NC23CC(NC(=O)CNC(C4(C(F)(F)F)CC4)=O)(C2)C3)ccc([N+](=O)[O-])cn1 c1(C(N2CC(COC)N(C(=O)Cc3cncs3)CC2)=O)cc(Cl)cc(C)c1N C1(OC)CC(OC(c2[nH]c(-c3cccnc3)nc2C)=O)CC(OC)C1 C(=O)(CN=c1cc[nH]cc1)N1CC2C(NC(C3CC34CCC4)=O)C(C2)C1 C1(OCCCF)CN(C(=O)COC2(CC(=O)NCCn3cccc3)CC2)C1 c1(CCN(CC(O)C(=O)N(CCC(=O)N(C)C)CCO)C)ccccc1N C1(NC(CCc2ccc(C)s2)=O)CC2CN(C(=O)CC(C)C)CCN2C1=O CC1=C(C(=O)N2CCC(C)(C(=O)NC3CC3C(C)(C)C)CC2)CCO1 N1(C(C2(CCC)CCC2)=O)CC(NC(C2CCCC2(F)F)=O)C(C(F)(F)F)C1 N1(C(C2(C(C)(C)C)CCC2)=O)CCN(C(=O)C(F)OC(F)(F)F)C(C2CC2)C1 Cc1cn(C)nc1C(=O)N(C)CC1(NC(=O)CCc2ncccn2)CC1 N1(C(c2cc(C)n(C(C)C)n2)=O)CCC2OCCN(C(C3CCC(C)O3)=O)C2C1 N1(C(C2CC3CC3N2C(c2ccc(Cl)c(Cl)c2)=O)=O)CCc2sc(Br)cc2C1 C(=O)(C1CCCc2cccnc21)NCC(C)NC(=O)C1=CCCCCC1 C1(C(=O)Nc2cccc(CCO)c2)CC2(CCN(Cc3sccc3Cl)CC2)C1 C1(CC(=O)NC(CCNC(C(C)(C)CC#N)=O)(C)C)Oc2ccccc2NC1=O Cc1nc[nH]c1CC(=O)NC1CC(C)(NC(=O)C(C)OCCC(C)C)C1 c1(C(=O)NC2C3(CN(C(CC(=O)OC)=O)C3)SCC2)ccc2c(c1)N(C)C(=O)C2 C(C(O)CN=c1cc(F)nc(S(C)(=O)=O)[nH]1)NC(C1C(C)(C)CC1)=O CC1CCCCN(C(c2cn(C(C)C)cn2)C(=O)NCCC2CC2)C1 Cc1cn2cc(CC(N3CCOC(c4ccc(F)cc4F)C3)=O)nc2s1 C=CCCC(CC(C)C)C(=O)N1CC(OC)C(NC(c2ccnc(F)c2N)=O)C1 Cc1ccn(CC(=O)NCC(C)CN(C(=O)CCCc2cnn[nH]2)C)c(=O)c1 c1(C(=O)NCCC2CCCN(C(CCC(=O)NC)=O)C2)sc(C#N)cc1Cl C12(CNC(C3(C)CCOC3)=O)CC(c3c(NC(=O)OC(C)(C)C)scn3)(CO1)C2 C(=O)(CC(C)(C)CC(F)(F)F)N(CCNC(c1c(C)c(Br)sc1)=O)C n1(CC(N2CCC3CN(C(C=NOC)=O)CC3C2)=O)c(C)nc2ccccc2c1=O CCCCCC(C)CC(=O)NCC1CCCC2(CN(C(=O)C(O)COC)C2)O1 CCCC(C#N)C(=O)N1CCC(C)(CNC(c2conc2-c2ccccc2)=O)C1 C1(C(=O)NC2C(NC(c3c(C)con3)=O)C2)CCc2c[nH]nc2C1 N1(C(C(CC)C)=O)CCC(CCN(C)C(c2coc(Cl)n2)=O)CC1 C1(N(C)C(c2cnnc(O)c2)=O)CC2CCC(C1)N2C(C1CC1(F)F)=O N1(N(c2ccc(CO)nc2)CC)CCCC(N(CC)CC)C1.c12nc(n[nH]1)NCC2 N1(C(CC(C=C)(C)O)=O)CCC(C(N2Cc3cncnc3C2)=O)CC1(C)C N1(C(c2cc(OC)no2)=O)CCC2CN(C(=O)C=Cc3ccncc3)CC12 c1(NC)cncc(C(=O)NC(CC2CC2)C(=O)NC2COC(C(F)F)C2)c1 C1(NC(C(C)CF)=O)CN(C(C2(C#N)CCCCC2)=O)CC2(CC2)C1 CCCCC(O)C(=O)N1CC(N(C)C)C(CNC(=O)C(=O)N(C)C)C1 C1(C(C(=O)NC(CC)C)N(C)Cc2cccnc2)CCC2(CC2)C1 c1(OCC)cc(C(=O)NC2CCC(NC(c3sc(OC)nc3Cl)=O)C2)oc(=O)c1 c1(CCCC(=O)NCC(CO)NC(CC2(C#N)CC2)=O)ccc(F)cc1 C1(CC(=O)NC2CCN(CCCNC(C3(CC(F)F)CCC3)=O)C2)CC1C1CC1 C(C(=O)N1CC(O)C(O)CO1)C1CCN(C(Cn2c(C)ccc2C)=O)C1 C1(O)(CNC(c2cn(CCCF)nn2)=O)CCCN(C(c2ccns2)=O)CC1 Cc1cc(C(F)(F)C(=O)NC2CN(C(=O)C=CC(C)C)CCC2F)cnc1Cl N1(C(C)CNC(c2ccnnc2)=O)CCN(C(C2(F)CCCC2)=O)CC1 c1(CNC(CC2C(C)(C)C(NC(=O)CC3CSC3)C2)=O)cccc2c1CCC2 N1(C(c2c(C)cco2)=O)CC2CCC(C1)N(Cc1ccc(F)c(OC(F)F)c1)C2 N1(C(CCC2CCCN(C(c3c(CC)c[nH]c3)=O)C2)=O)CC2CCCCC12C N1(C(C2CCN(C(CC)=O)C2)=O)CCCC(NC(c2cscc2OC)=O)C1 C=C(Cl)CCC(=O)N1CCOCC1CN(C(=O)CCSc1ccccc1Cl)C C1(NC(c2cc(F)ccc2F)=O)CCN(C(c2csc(Cl)c2)=O)CC1F CC(=Cn1ccnn1)C(=O)NCCCC(C)NC(C1SCCS1)=O C1(CC)(NC(=O)C(C)OCOC)CCN(C(=O)C=CCF)CC1 C1(C(N2CCC(CCNC(C34CCCN3CCC4)=O)C2)=O)C(F)(F)C12CCC2 C=CC(F)(F)C(=O)NC1CC(NC(c2csc(O)n2)=O)C1 n1(CC(N2CCC(NC(C3C(C)C3)=O)C2(C)C)=O)nnc2c1CCCC2 C1(NC(C(CCC)=CCC)=O)CC2(CCN(C(C3(C)CCCS3(=O)=O)=O)C2)C1 c1(CNC(c2cccnc2)=O)ccnc(C(=O)NC(CC2CCCC2)CO)c1 c1(CC)ccc(OCC(=O)NC2CCC(C(=O)Nc3ccc(C)cc3)CC2)cc1 CCC(CC)C(C(=O)N(CC(=O)NC1CCC(C(N)=O)C1)C1CC1)OC C#Cc1ccc(C(=O)NC2CC3(C2)CC3NC(c2cnc(C)[nH]2)=O)c(OC)c1 N#Cc1cc(C(N2CCN(C(C3CCc4nnnn4C3)=O)CC2)=O)c(O)cc1N C1(CC(=O)NC(C2(O)CCCCC2)C(=O)NCc2c(C)ncs2)CC2C=CC1C2 CP(C)(=O)CCC(=O)C1C(C(=O)N(c2c(O)cccc2F)C)C(NC)C1 CCC(C)CCCCC(=O)N1CC(C)(C)CC1CC(=O)Nc1cnc(Cl)c(C)c1 C1(C)(NC(C2(C)N(C(c3cc(C)n(C)c3C)=O)CC(O)C2)=O)CN2CCC1CC2 C1(CC(=O)NCCO)CC(O)C1(C)C.n1(CCN(C(C)=O)CC)cc(C)nn1 Cc1ccc(O)c(C(=O)NC(C)CCNC(c2cccnc2Cl)=O)c1 c1(C(CN(C(=O)CN(CC(C)(C)C)C)C)NC(COC(C)=O)=O)ccccc1 CCCC(C(=O)N=c1ccn(C(F)F)[nH]1)NC(=O)CN1CCCC1C Cc1ccc(C(=O)NC2CN(C(=O)CSc3n[nH]c(=N)s3)CC2C)c(F)c1 S(=O)(=O)(c1c[nH]c2cnc(Cl)cc12)NC(c1ccc(N2CCOCC2=O)cc1)=O c1(C(=O)NC(C(C(C)C)NC(c2c(OC)nsc2)=O)C)c(O)ncc2c1CCC2 C1(CN(C(=O)C(F)n2cccn2)CC)CCC(NC(CC2C(CC)C2)=O)CC1 CC(c1ccco1)=CC(=O)NCCCC1CCCN1c1ccnc(C2CC2)n1 c1(C(=O)NC2C(C(NOCC)=O)CCOC2)cc(F)ccc1O c1(C(=O)NCCC(O)C(=O)NC2(c3ccccc3)CC2)ccc2cc[nH]c2c1 N1(C(C2CC3CCC2CC3)=O)CC2CC(NC(C3(n4nccn4)CC3)=O)CC2C1 C1(C(=O)NCCN(C(CN(C)C)CC(C)C)CC)CCCC2C1C2(F)F C1(CC)CCCCCCN1C(=O)COC1CCN(C(c2ccc(F)c(F)c2)=O)C1 CCC(C)C(O)CC(=O)NC(CC)CCCC(=O)NC(c1cnn(C)c1)C C1(NC(c2c(CCC)nns2)=O)CCC(C)(CNC(c2ccc[nH]2)=O)C1 Cc1cc(C)nc(N2CCN(C(c3cccc(O)c3)=O)CC2CO)n1 c1(C(N2CCCC(NC(C3(CC=C)COC3)=O)C2)=O)cc(S(N)(=O)=O)c[nH]1 c1(C(C)NCc2c(NC)nccc2)ccc(F)c(Br)c1 C12(NC(C(CC)F)=O)CC1CN(C(c1cncc(-c3ccccn3)c1)=O)C2 N1(C(c2sccc2Cl)=O)CC2CC(C1)N(C(c1nc(C3CC3)ncc1Cl)=O)C2 Cc1nn(C)c2c(NC(C)CS(C)(=O)=O)nc(=NC(C)c3ccncc3Cl)[nH]c12 N1(C(CCCC=C)=O)CC2CCCCC2(NC(c2nc(OC)c(C)s2)=O)C1 C=CCC(C(=O)N(C1CCN(C(=O)C(CCCC)ON=C(C)C)CC1)C)C(C)C n1(C(CC)C)nnnc1C(CCC1CC1)NCc1cocn1 C1(NC(c2ccn(CCF)n2)=O)C2CN(C(C3(F)CCCOC3)=O)CC12 c1(C(N2CCC(O)(C(=O)OC)C2)C(=O)NC(CC)C)cc(S(C)(=O)=O)c(C)o1 c1(NC(CNC(CCOC)CNC(=O)Cc2cocn2)=O)c(N)cccc1F c1(C(N2CC(CC=C)(C(=O)NC(CC3CC3)CO)C2)=O)cc2ccccc2[nH]1 N1(C(C2(C(C)C)CCN(C(=O)C(F)n3ccnc3)C2)=O)C2CCCC1COC2 c1(SC)nc(=NC2CCCN(C(=O)CC34CCCN3CCC4)C2)c(C#N)c[nH]1 Cn1nc(Cl)c(C(=O)N(CCCN(C)C)CCNC(C2C3CCCC23)=O)c1Cl c1(OC)c(Cl)ccc(Cl)c1C(=O)NC1CC(CNC(C2NC(=O)CC2C)=O)C1 CN1Cc2ccccc2C(NC2CCCC2CN=[N+]=[N-])C1 CCC(CC(=O)Nc1cnccc1CO)NC(c1cc(C)[nH]c1C)=O C=C(C)CC(C)C(=O)N1CCN(C(=O)C=CSC)CC1CCOC CCCCCCC(CC)C(=O)NC(C)CNC(c1cncc(NC)c1)=O C1(CC=C)(C(=O)NCCC2(O)CN(C(c3cc(C(C)C)on3)=O)C2)CCOCC1 N1(C(CN(CC)CC)=O)CCC(n2cc(Cn3cc(C)cn3)nn2)C1 Cc1ccc(C(=O)N(C23CC(Br)(C2)C3)C(=O)CN2CCCCCC2COC)c(C)c1 C1(CNC(=O)OC(C)(C)C)OCCC1(C)C.C12C(C1(C)C)NC2=O C(=O)(C(C)(CO)NC(=O)C(c1cccn1C)=O)N1CC(CS(C)=O)C1 C(C(F)(C(=O)NC1COCCC1CO)C(C)C)NC(c1c(C)scn1)=O Cn1cc(NC(=O)CC2(C)CCN2C(=O)Cc2cnns2)cn1 C1(C)(CNC(C2CCC3CC23)=O)CN(C(C2(OC)CC(C)C2)=O)CC1C C(C)(C(C(=O)NCC1OCCC1(C)C)C(C)C)NC(c1c(NC)nccc1)=O C(C)(C)(CN=c1[nH]cnc(NCc2cccnc2C(F)(F)F)c1C)OC c1(C(=O)NCc2scc(C(=O)NCC(CC)C(C)C)c2)ccc(C)c(C)n1 c1(CCC)ncoc1C(=O)N(CC(=O)NCC(=O)NCC=C1CCSCC1)CC Cc1ccc(C(=O)N(CC(N2CCC(OC(C)=O)C2)=O)C2CCC2)c(O)c1 c1(OC)cnc(C(N2CC(CNC(c3ccnc(C)n3)=O)C3(CC3)C2)=O)c(F)c1 C#CC1(O)CC(C(=O)NCC(O)C(=O)NCCN2CCC3CC23)C1 C(=O)(C(F)C(C)CNC(C1CC(F)CN1C)=O)NC(C(C(=O)OC)C)C CC1CCCC(N(C(C2(NC(=O)CNC(=O)C(C)(C)C)CC2)=O)C)C1 c1(C(=O)Nc2c(C(=O)NCC)cccc2)nccc(C#N)c1Cl C1(C)(N(C(=O)CCOC2CN(C(=O)CC3C=CCC3)C2)C)CCOCC1 CCCCC(O)C(=O)N1CCC(C)(C)C1CNC(=O)CCc1ccc(CC)cc1 c1(C(=O)NCC(C)N(C(c2ccc(C(N)=O)s2)=O)CC)ccc(C2CC2)cc1 Cc1c(CC(=O)NCC2(C(N3CC(CO)C(CO)C3)=O)CCC2)cnn1C C1(NC(CC2(OC)CCCC2)=O)CN(C(=O)C(C)N=[N+]=[N-])CC1O C1(NC(CC(=C)Br)=O)CC2CC(C1)N(C(c1cccc(N)c1F)=O)C2 Cc1cn(C)cc1C(=O)NCCN(C(c1ccc(N2CCCC2)nn1)=O)C(C)C C(CSC(C)Cn1cnnc1)(C(=O)NC)NC(CC=CC=C)=O C1(N(C(c2nc(C#C)sc2)=O)C)CCCN(C(C2CC2(Cl)Cl)=O)CC1 c1(C(N(C(C)C)CCNC(C2(C(F)(F)F)CC2)=O)=O)ccc2c(n1)CCC(C)C2 c1(OC)ccc(CC(N2CCN(C(c3oc(C)nc3C)=O)CC2C)=O)c(Cl)c1 c1(C(=O)NCCCNC(c2c(COC)scc2)=O)ccc(F)c(F)c1F N1(C(c2c[nH]c(=NC)o2)=O)CCC2(CC1)C(OC)CC2NC(c1ccc(C)o1)=O c1(C(N2C(CNC(CCOC(C)=O)=O)CCC2)=O)cc(C(C)C)nn1C c1(CNC(C2C(C)(C(C)C)C2)=O)ccc(C(=O)NCC=CCl)cn1 C1(CC)CN(C(C2CC2c2sccc2C)=O)CCN1C(=O)C(=Cc1c[nH]cn1)F Cc1sc(C(=O)NC(C)CN(C)C(C2(O)CC(CF)C2)=O)cc1[N+](=O)[O-] O=C(C1Cc2ccc(F)cc21)NC1CCN(CC(N2CCOCC2)=O)C1 C(=O)(C(C(C)C)C1CCC1)NC(C(=O)NCC(=C)C)Cn1ccnn1 C1(NC(=O)NC(C2CCCCO2)CC)CCC(OCC2CC2)CC1 C(CNC(=O)CN1CCSCC1)(C(C)(C)C)NC(C(CC)Oc1ccccc1)=O c1(NC)cc(Cl)ccc1C(=O)NCCC(C(C)C)NC(c1cc[nH]n1)=O C1(NC(C=C2CCN(C)CC2)=O)CC2CC1CN(C(C1CCC(O)CN1C)=O)C2 C(=O)(CC(C)CN(C)C)NC1(C)CC(NC(CC2CC(OCC)C2)=O)C1 c1(CCN=C(NCC2(C#N)CC2)NC2CC2)ccc2c(c1)OCCO2 CCCC(CC)C(=O)NC1CCC(F)(CNC(=O)Cn2ccc(C3CC3)n2)C1 C(=O)(C(C)C(O)C(C)C)NCCOCCN(C1CCCC1)CCO.CC(C)C1C(=O)N1 Cc1ccc(CC(=O)NCC2COC(CNC(c3ccn(C)n3)=O)C2)cc1Br C1(NC(c2cccnn2)=O)CCN(C(C2(O)CCSC2)=O)CC1CO N1(C(=O)Cc2cnccn2)CCC12CCCN(C(C1CC(O)C1)=O)C2 C1(C(N(C)CC2N(C(CC(C)(C)OC)=O)CC(F)C2)=O)CCc2c[nH]nc2C1 c1(C(CNc2c(NC(CCc3cc(C(=O)OC)c(C)o3)=O)c[nH]n2)=O)cc(F)cc(Cl)c1 C(=O)(C1=NOC(CNC(C2CCCSC2)=O)C1)N1CC(CC)C1 C1(C(N(C)Cc2cnn(-c3ccccc3)n2)=O)CCCCC1NCCO C1(NC(c2c(CC)onc2)=O)CC2CC(NC(=O)CCCc3csc(=N)[nH]3)CC12 c1(C(N2C(CN(C(C(C)NC(CC)=O)=O)C)COCC2)=O)cc(F)c(F)cc1Cl C(c1ccn(C)c1)=CC(=O)N(CCN(C(c1c(SC)ccs1)=O)C)C C1(NC(c2cc(Br)c[nH]c2=O)=O)CCN2CCCC2C1 N1(C(c2n(C)ncn2)=O)CCC2(CC(NC(c3cnn(C(F)F)c3)=O)C2)C1 CCCCC(C(=O)N1CCCC1(C)CNC(=O)C(C#N)C1CC1)NC(N)=O C=Cc1ccc(C(N2CCOC(C(=O)NCCOCC3CCC3)C2)=O)cc1 S(=O)(=O)(c1cnccc1N1CCCC2(CCOC2)C1)N1CCCC(C#N)C1 N1(C(c2scnc2C(F)(F)F)=O)CC2CCCC(C1)N2c1ncc(Br)c(O)n1 C1(NC(=O)CN2CCN(CCc3ccsc3)CC2)CCc2c[nH]nc2C1 c1(C(=O)NC(CN(C(C2CCC(=O)N(C)C2)=O)CC)C)cnc2c(C)nsc2c1 CC1CCN(c2nccnc2F)CC1NC(=O)C(C)(C)N1CCCCC1 c1(C(=O)NCCc2ccn(CC)n2)cc(F)c(F)cc1Cl Cc1coc2c(C(=O)Nc3nc4ccc(O)cc4s3)cccc12 Cc1ccc(C(N2CCC2C(=O)NCC2CCC3(CC2)CC3)=O)c(O)n1 c1(SC(C)C(=O)NCC(CO)NC(c2cnc(O)s2)=O)ccccc1Cl N1(C(=O)CN2CCCC2=O)CC2CCN(C(c3ccc4nsnc4c3)=O)C2C1 C1(CCCC)CCCN(C(C2CN(C(C3C=CCS3)=O)CC2F)=O)C1 c1(SC)cccc(-n2nc(-c3cccc(OC(C)(C)C)c3)nc2C2C(C)C2C)c1 n1(CC)nc(C(=O)NC2CC2C(=O)N=c2cccn[nH]2)c2ccccc12 C(C(F)C(=O)N(CC)Cc1ccoc1)C1CN(C(C(C)=CC=C)=O)C1 c1(NC(C2CC(NC(c3ccnc(F)c3Cl)=O)C2)=O)c(Cl)cnnc1Cl CS(=O)(=O)c1cc(C(N2CCC(NC(=O)Cc3c[nH]c4cccnc34)C2)=O)co1 N1(C(C=C(C)C)=O)CC2COCC2(C(=O)NCc2c(C)cccc2C)C1 C(=O)(C(O)CC(C)(C)C)NCC(CC)NC(C(C)SCCCC)=O N1(C(c2scc(C#N)c2)=O)CCOC2(CCN(C(c3ncncc3Cl)=O)CC2)C1 c1(C(=O)NC2CN(C(c3cc(F)cc(Cl)c3)=O)CC2F)csc2c1CCCC2 C1(C(N(C2CCCOC2)CC)=O)CN(C(=O)C=C=C(C)C)CC1C C12(CNC(=O)C=Cc3ccoc3)CC1CN(C(=O)CCOc1ccccc1F)C2 c1(OCCN(CC(CN(C(C(C)=CCC)=O)C)O)C)nnnn1C1CCCC1 c1(OC)cc(C(=O)NC2(C)CCN(C(=O)C(F)C3CC3)CC2)c2ccccc2n1 CC1CN(CC(=O)NCC2CCCO2)CCN1c1cc(N(C)C)ncn1 N1(C(=O)Cc2ccsc2)CCCC2(CCN(C(C3CCCN4CCCC34)=O)C2)C1 C1(NCCS(=O)(=O)NC(C)C)CCN(N(C(C)=O)C(C2(SCC)CC2)=O)C1 N1(C(c2cncc(OCC)c2)=O)CCCCC(NC(=O)C(C)n2cccc2)C1 c1(C(=O)NC(C)CNC(=O)C(c2cncc(F)c2)C)cc(C(F)F)cc(F)c1 c1(C(N2CC(F)CC(NC(=O)CC(F)(F)F)C2)=O)cccc2cnccc12 c1(NC(C2CCC(NC(C3(COC)CC3)=O)C2)=O)cnc(C)c(Br)c1C S(=O)(=O)(c1cccc(F)c1F)NC(CNCCC(N)=O)=O C1(CCOC)CCN(C(=O)C(C)CN(C(=O)C(C)CO)C)C1 c1(C(=O)NCC(C2CC2)NC(CCCOC(C)=O)=O)nc2cccnc2s1 c1(OC)ccc(S(=O)(=O)N2CC3C(C(=O)Nc4cc(C#N)c(Br)cn4)C3C2)cn1 C1(NC(C2CC2(F)F)=O)CCCN(C(=O)CSC2CCOC2=O)CC1 S(=O)(=O)(c1ccc(NCc2cnsc2)c(C#N)c1)N(CC(C)C)C1CCC1 N1(C(C2(CCNC(C=CC(CC)C)=O)CC2)=O)CCC2(CCCO2)C1 Cc1cc(C(=O)N(CC(C)N(C(=O)CC(C)(C)C)CCC)C)c2c(c1)CCC2 c1(CC)ccc(C)c(C(N2CCN(C(=O)Cc3cccc(F)c3)C3CC23)=O)c1 CCC(C)CC(=O)NC1C2CC1N(C(=O)C(C1CCCC1)OC)C2 C1(NC(c2sccc2CO)=O)CCCC1NC(C1CC1c1ccccc1)=O c1(CC(N2CCC(CCNC(CCC=C)=O)CC2)=O)ccc2c(c1)CCN2C c1(C(N2CCC(NC(c3ccc(COC)s3)=O)C2C)=O)ccc(F)c(F)c1 C1(CC(=O)NC2(CN(C(c3cc(C)sc3)=O)C)CC2)CC2(C1)CC1(CCC1)C2 CC1=C(C(=O)NCC2CCN2C(c2cn(C)nc2OCC(F)(F)F)=O)SCCO1 C12(C(=O)NCC(CC)NC(=O)C(C)=C3CCC3)CCC(n3cnnn3)(CC1)C2 CC(C)C(CNC(=O)Cc1nccn1C)NC(c1ccoc1C(F)(F)F)=O N1(C(=O)C(F)C2CCOC2)CC(F)(F)c2ccccc21 c1(C(N2CCC(F)(F)C(CNc3ncccn3)C2)=O)coc2cc(O)ccc12 c1(C(N2CCC(NC(Cc3c(C)noc3)=O)(CO)C2)=O)cc(=O)n2ccsc2n1 c1(C(=O)NCCCC2N(CC(=O)N(CC)CC)CCC2)cn2nccc2nc1C C1(N(C(COC(C)=O)=O)C)CCC(NC(=O)C(F)CC2CCOC2)CC1 N1(C(C2(c3ccc(Cl)c(F)c3)CC2)=O)CCC2(CC1)OCc1ccccc12 Cc1cc(F)c(C(N2CCOC3(CCC3)C2)C(=O)NC2CCOC2)nc1Br c1(C(=O)NCC(CO)NC(C(C(=O)OC)C)=O)c(C)nn(-c2ccccc2)c1C N1(C(CC)C)CC(C(N2CCN(CCN(C)Cc3ccccc3)CC2)=O)CC1=O CCC(C)CC(C(=O)NCC(C)COC)NC(=O)CCN1CCCCC1 C(C)(C)(C(=O)NC1CC(CCNC(C2CC2c2cccnc2)=O)C1)OC(C)C#N C1(C(N2CC(NC(=O)C3=CSCS3)C3(C2)CC3)=O)Cc2ccc(F)cc2C(=O)O1 N1(C(C(C)N(C)C)=O)CCC(C(=O)C(C)(C)C)CC1 CC1(C)CCC(F)(F)CC1C(N1CCCCCC1CNC(=O)C(=O)NC1CC1)=O CC1CCC(C)(NC(C2CC(C)N2C(C23CC(C#N)(C2)C3)=O)=O)C1 C1(CC=C)(NC(=O)CCCCCC)CC2CCC(C1)N2C(c1n[nH]c(SC)n1)=O c1(C(=O)NC(C)CN2CCN(C(=O)CSCC(N)=O)CC2)cccc(F)c1F C(C(CC(=O)N1CC(O)(n2cnnn2)C1)OC)NC(C(CC)n1ccnc1)=O N#CC1(C(=O)NC2CCCCC2CNC(=O)CC(F)(F)F)CC2CCC1CC2 CC1(C(=O)NC2CC(C(=O)NCC(O)Cc3cnc[nH]3)C2(C)C)CCOCC1 C1(NC(c2cc3c([nH]2)CCCC3)=O)C2CC3CN(C(=O)C=CBr)C1C3C2 C1(CNC(C(C)NC(CC)=O)=O)CC2COCC2N1C(c1ccc(N)cc1Cl)=O CCC(C)(CNC(=O)COC)NC(c1cnn(CCC(F)(F)F)c1)=O C1(CC(=O)NC2CC(OC(F)F)C2)CCCN(c2cc(O)ncn2)C1 C1(NC(Cc2ccn(C(C)C)n2)=O)CCCN(C(=O)C(F)Cc2ccccc2)C1 c1(C(C(N2CCC(CN(c3oc(C)cc3C)CC)C2)=O)(C)O)ccc(F)cc1 Cn1cc(C(N2CCCC2C2(NC(=O)C=Cc3cn[nH]c3)CC2)=O)c(O)nc1=O Cc1cc(C(=O)NCC(CO)NC(c2csc([N+](=O)[O-])c2)=O)c2cnccc2c1 c1(CCC)c(C(=O)NCCCN(CCC)C(C2CC3(CCC3)C2)=O)nnn1C C1(C)(C(N(C(CNC(c2c(CC)ccs2)=O)C)C)=O)CCCCNC1=O N1(C(C(CCCC)O)=O)CC2CCC(C1)N2C(C1(C)CC2CCC(C1)S2)=O N1(C(c2ccc(C(=O)OC)s2)=O)CCC(NC(=O)CN2CCSCC2)C(C)(C)C1 C1(CS(=O)(=O)NC(c2ccc(C3CC3)cc2)C(F)(F)F)CCC2(CCC2)OC1 Cc1ccc(I)c(C)c1NC(C1CCC2(CN(C(=O)Cn3cccn3)C2)O1)=O CN1CCN(C(=O)C(C2CCCCCCC2)O)CC(O)C1 C(=O)(C(C)CCC(C)(C)C)NCC(CC)N(C)C(c1ncn(CC)n1)=O CC1CN(C(=O)CSc2cccc[n+]2[O-])CC1CNC(=O)C=CC1CCOCC1 c1(C(=O)NC2C3CN(C(c4cc(C)sc4C)=O)CC32)[nH]nc([N+](=O)[O-])c1Cl CC1(C)C(NC(=O)C=Cc2ccncc2)CCN1c1ncc(C(F)F)cn1 N1(C(=O)C2=NOCC2)C2CCC1(c1nn[nH]n1)CC2 C1(C(=O)N(c2cc(Cl)ccc2F)CCO)CC(F)CN(C(c2ccccc2)=O)C1 c1(C(N(CCN(C(C2CC(C(=O)OC)C2)=O)CC)CC)=O)ncc([N+](=O)[O-])n1C c1(CC(=O)NC2CN(C(CC3ON=C(CC)C3)=O)C2)cc(OC)ccc1OC c1(C(N2CCCC(NC(CC(C)C)=O)C2C)=O)coc(C#Cc2ccccc2)c1 C(=O)(C1CCCn2nccc21)NC1CC2(CCCN(C(C(C)NC(C)=O)=O)C2)C1 N1(c2nc(C)nn2C2CC(C)CC(C)(C)C2)CC(C)(C)c2ccccc21 N1(C(C=CC)=O)CC(CNC(C2(C(F)(F)F)CCC2)=O)CC1(C)C C(=O)(C#CC(C)(C)CNC(C1(CF)CCOCC1)=O)NCC(C)OCC=C c1(NC2C(C)(C)CN(C(=O)CCn3cncn3)C2)cc(C(F)F)nc2ncnn12 C12(OC)CCC(C(=O)NC(C)CC3CCN(C(=O)C4CC4)CC3)(CC1)C2 c1(SC(C(=O)NCCC(CNC(CNC(CC)=O)=O)O)C)ccc(C)c(C)c1 C1(C(N2CCC(O)(CN(C(CC(C)C3CC3)=O)C)CC2)=O)OC(C)(C)OC1(C)C Cc1noc(CCC(=O)NC(C)C(CO)NC(=O)C(N2CCOCC2)C)n1 CC1=C(C(=O)NC2C3CCN(C(=O)CC4C=CS(=O)(=O)C4)C23)SCCO1 C1(C)(CNC(C2(CO)N(C(CCc3cc(C)no3)=O)CCC2)=O)CCN(C)CC1 CCC1=NOC(CNC(=O)C(C2CCCC2)NC(=O)Cc2cc[nH]n2)C1 c1(C(NNC(=O)C=Cc2ccccc2F)=O)ccc2c(c1)OCCNC2=O CCC(C)C(O)CC(=O)N1CCC(C(=O)NC(C)C(=O)N(C)OC)C1 c1(C(N(CCCN(C(=O)Cn2[nH]cnc2=N)C)C)=O)nn(C)cc1Cl C12(CNC(=O)CCc3ccc(Cl)cc3)CC1CN(C(C1CCS(=O)(=O)N1)=O)C2 C(C1c2ccsc2CCN1C(=O)Cc1cn[nH]c1)NC(C1CC1n1nccn1)=O N1(C=O)CCN(C(c2ccc(COC)s2)=O)CC1.C(=O)(CC(C1CC1)SC)NCC N1(C(Cc2ccc(C)o2)=O)CCC(O)(CNC(=O)CCOCC2CC2)CC1 c1(CC(N2CC(C)(C(=O)Nc3ncccc3CO)C2)=O)cc(C(F)(F)F)cc(F)c1 C1(C(=O)NCC2CC(C(=O)NCCOCCOC)C2)CC2C=CC1O2 c1(CN(C(CC2(N(C(C3C(C)(COC)C3)=O)C)CC2)=O)C)nnnn1C c1(CC(C)(C)C)ncc(C(=O)OCCNC(C2CCC2)=O)o1 c1(CC)ccc(C(=O)N(C(C)CNC(=O)CC(O)C2CC2)C)c(F)c1 C(=O)(C(F)(CC)C(=O)OC)NC1CC(NC(c2ccc(CSC)o2)=O)C1 N1(C(C(CCOCC)NC(c2ccc(F)c(O)c2)=O)=O)CCC12CCCSC2 C=CC1(CC(=O)Nc2ccccc2-c2ncc[nH]2)CCCCC1 C1(CNC(c2c(C)n[nH]c2)=O)COC(C)(C)CN1C(c1cnn2cnnc2c1)=O CC1CC(C(N)=O)c2ccccc2N1C(=O)CC1OCc2ccccc21 N1(C(CCCC(CC)C)=O)CC2CCCCC2(NC(=O)C=C2CCC2)C1 N1(C(c2c(C)ccc(C)c2)=O)CC(C)CN(C(c2ncc(Cl)cc2Cl)=O)CC1C C(CO)(C(=O)N=c1ccn(C(C)CC)[nH]1)NC(c1ccc(CC)cc1)=O N1(C(c2cn(C)nc2CC(C)(C)C)=O)CC2(CCCC2N)C1 c1(OC(C)C)cccc(C(=O)NC2C3CC2N(C(c2nccn2C)=O)C3)c1 C(=O)(C#CC1CCCCC1)N1CCC(CN(CC(=O)NCCC)C2CC2)CC1 N1(C(c2ccc(C)s2)=O)CCN(C(C2CC(=O)N(c3cn[nH]c3)C2)=O)CCC1C N1(C(C2C(C(C)(C)C)CC2)=O)CCCCCC1C(N1CCC1C(N)=O)=O C1(C(N(CC(C)SC)C)=O)CC(N=[N+]=[N-])CN1C(=O)Cc1csnc1C c1(OC)cc(C(=O)NCCN(CC(C)O)C(C2CC2C)=O)cc2c1OCCO2 c1(C(=O)NCC(CO)NC(C(c2scc(C)n2)(F)F)=O)cnc2cccnc2c1 C(=O)(C1CCCc2nnn(C)c21)NCCC1CC(NC(C=C(C)Cl)=O)C1 c1(CC)ccc([N+](=O)[O-])cc1S(=O)(=O)NNC(=O)C(N)COCc1cccc(C)c1 N1(C(C2C(C(C)C)OCC2)=O)CC2CC1C2C(=O)NCC1CCCCN1C CC1Oc2ccc(CN3CCCC(CCNC(=O)C(O)C(C)(C)C)C3)cc2C1C C1(CCC(=O)NC(C)CCN(C)C)CCN(C(C2(C#N)CC2(C)C)=O)CC1 c1(C(N2CC(C)(CNC(C3N(C)CCC3)=O)C2)=O)ccc2ocnc2c1 CCC(C)C(C(=O)NCC1CC(NC(c2cn(CCN(C)C)nn2)=O)C1)OC Cc1ccc2c(c1)SC(C(=O)NC1CCC1NC(=O)C(C)(C)c1nncn1C)C2 C=CCC(C(=O)NCC(C1CC1)NC(=O)CCN(C)CC)C(C)C c1(N(C2CN(C(C34CC(C)(CO3)C4)=O)C2)C)cc(C(N)=O)ccc1[N+](=O)[O-] c1(C(=O)NC(c2nc(C)cs2)CC)ccc(Cc2cncc(F)c2)cc1 CC1(C(=O)NCC(CC2CCCC2)CO)CCN(C(=O)CC2(O)CCCC2)CC1 C1(NC(=O)CCOC2CN(C(C3OCC4CCCC34)=O)C2)CN2CCC1CC2 C12(C(N3C(CNC(c4ccc5c(c4)CC5)=O)CCCC3)=O)COC(CCO1)C2 C1(NC(c2cc(C3CC3)cnc2Cl)=O)CC2CCC(C1)N2Cc1cncc(Cl)c1 C1(NC(=O)CCc2ccc(F)cc2)CC(O)CN(C(c2[nH]cc3c2CCC3)=O)C1 C1(NC(c2c(CC)nco2)=O)CN(C(c2ccnc(OC)n2)=O)C2(CCOC2)C1 c1(C(N(CCC)CCNC(C2(S(C)(=O)=O)CC2)=O)=O)ccnc2ncc(C)cc12 c1(CC)cc([N+](=O)[O-])ccc1N1CCN(CCNC(=O)CC2CCC(C)C2)CC1 Cc1[nH]nc2ncc(C(=O)NC3CCC(C)N(C(=O)CCC4CC4(F)F)C3)cc12 c1(SCC(=O)NCCSC)c(C)cc(C)cc1Cl.C1(C)C(=O)N1CCC c1(C(=O)NCCC2(NC(C3CC3Cl)=O)CCOCC2)c[nH]cc(Cl)c1=O c1(CCC(=O)N(C2CN(C(c3cscc3F)=O)CC2F)C)ccc2c(c1)CCO2 C(=O)(C(C(C)(C)C)OC(C)C)N1CC2C(NC(c3ccn(CCC)n3)=O)(C2)C1 C1(OC)CCCCN(C(C2CC(=O)C2C(C)(C)C)=O)C1.c12c[nH]c(c1)NC2=O C(CN=c1[nH]c(=NC2C=CC(CO)C2)[nH]c2c1CSC2)(c1ccccc1)N(C)C C1(OCC(=O)OC(C)C)CCC(C)N(C(c2cn(CC(=O)CCC)nn2)=O)C1 N1(CC)CC(C(=O)NC2CCCC(NC(=O)CCc3cnc[nH]3)C2)CCC1=O N1(C(C(C)(C)SC)=O)Cc2[nH]nc(C(=O)NCc3cc(C)co3)c2C1 Cc1csc2ncnc(N(CCC3CCCNC3)Cc3c(Cl)ccc(Cl)c3F)c12 Cc1ccn2cc(C(=O)NC3CN(C(c4ccc(F)cc4Cl)=O)CC3C)nc2c1 CC(N=c1cc[nH]cc1S(=O)(=O)N(C12CC(C1)C2)C)C1CN(C)CCO1 N1(C(c2c(C)ncc(Cl)c2)=O)CCN(C(=O)Cc2ccns2)C(C)C1C C1(N(C)C)CCN(C(=O)C(CC2CC2)NC(=O)COC2CCCCC2)CC1 C1(NC(c2cc(Cl)c(F)c(Cl)c2)=O)CN(C(=O)CC2CCOCC2)CCC1(F)F N1(C(C(CCC)O)=O)CCN(C(c2ccn(C(C)C)n2)=O)CC1C C=C=C(C)CC(=O)NC(C)(C)CNC(C1(N(C)C(=O)OC(C)(C)C)CC(O)C1)=O C1(NC(CC)=O)C=CCC(C(N2CCC(C(C)CO)CC2)=O)C1 N1(C(c2cccc(C)c2N)=O)CCC2(C1)CN(C(C1(C)CC1(F)Cl)=O)CCO2 C(=O)(C(C)(F)C(=O)NCC1CCN(C(c2csc(-c3cnccn3)n2)=O)C1)OC CC(C(=O)NCc1cccnc1CNC(=O)C(CO)N(C)C)S(C)(=O)=O c1(C(=O)NC2CCC(CCNC(C3(CC=C)CCC3)=O)C2)ccc(C)cn1 C1(N(C(c2c(CC)onc2)=O)C)CN(C(=O)Cn2cc(C)cn2)CCC1C c1(C(=O)NC2CC3CN(C(C(=O)N(C)C)=O)CC32)c[nH]c2nccc-2c1 C(CCCCCN(C)C(c1ccco1)=O)NC(C1C=C(C)CS1)=O C(C)(N=c1[nH]c(=N)[nH]c(=NC(C)CCC2CCCC2)[nH]1)c1cccc(SC)c1 C12(C(=O)NCCC3N(C(c4n(C)ccn4)=O)CCCC3)CCOC1CC(=O)NC2 N1(C(C2C(OCC)C2)=O)CC(N=c2[nH]c(Cl)ncc2[N+](=O)[O-])CC1C N1(C(C2(OC)CCCOC2)=O)CC(C(=O)NCC2CC2C(C)C)CC(C)C1 N1(C(CCC(=C)C)=O)CCC2(CCC(NC(C3(Cl)CC3(F)F)=O)C2)CC1 N1(C(C(C)SCCCC)=O)CC2CCN(C(=O)COC(C)C)CCC2C1 N1(C(C(CN(C)C)N(C)C)=O)CC2(C)CC1(C(=O)NCCC1COCCO1)C2 C=CC1(C(N2CC3C(CNC(c4cccc(C)c4Cl)=O)C3C2)=O)CCCCC1 n1(NS(=O)(=O)c2cccs2)c(-c2ccc(C(=O)OCC)cc2)nc2ccccc12 C(C(C(=O)NC(c1cccnc1C)C)C(C)C)NC(C(C=C)(C)O)=O c1(SCC(C(=O)NC(CNC(c2cn(CC)nc2)=O)C2CC2)C)ccc(F)cc1 CC(C(C)C)=CC(=O)NC(C)(C)CNC(=O)CCC1CC1(F)F c1(C(=O)NCC2(C)N(C(C3N(CC)CCOC3)=O)CCC2)nc(C)ccc1OC c1(C(=O)NC(C(=O)N(C)CC2(O)CCC2)Cc2cn[nH]c2)ccc2c[nH]nc2c1 Cc1cnc(Nc2ccc(C)c(C(N3CC(N(C)C)C3)=O)c2)nc1C n1(CC(=O)NCC(CNC(=O)C=CCCc2ccccc2)O)cccnc1=O N1(C(c2cccc(C)c2)C(=O)Nc2ccccc2)CCS(=N)(=O)CCCC1 Cc1ncc(Cl)c(C(N2CCN(C(=O)CN(C(=O)C(C)CC(F)F)C)CC2)=O)n1 Cc1sc(N)c(C(N2CC(NC(=O)C(C)Cc3ccco3)CC(C)C2)=O)c1C c1(CC(=O)NC2(CCNC(=O)CCc3cnc[nH]3)CCC2)ccc([N+](=O)[O-])cc1 CC1(C)COC(=O)C1NC(=O)CCCn1cc(CC2CCCOC2)nn1 c1(C(=O)NCCn2ccc(C(=O)NC(c3nc(C)sc3)C)c2)cncc(C#N)c1 c1(C(=O)NC(C2N(C(C(C)NS(C)(=O)=O)=O)CCC2)C)ccccc1CCN(C)C C=C(C)CCC(C)NC(C1CCC(NC(=O)CC2CC(=O)C2)C1)=O Cc1ccc(C)c(C(=O)NC2COCCN(C(=O)C(c3ccc(O)cc3)=O)C2)n1 N1(C(c2ccc(CSc3c(F)cccc3Cl)o2)=O)CC(C(=O)OC)CC(F)(F)C1 Cc1cccc(C(=O)NC2CC(CCNC(c3cn(C(C)C)nc3C)=O)C2)c1C c1(N2CCCC(NC(C3C(C)OC(C)C3C)=O)C2C)cc(C#N)ccc1[N+](=O)[O-] N1(C(c2c(C)nc(CC)o2)=O)C2CC=C(C(=O)NCCOC3CCOC3)C1CC2 N1(C(c2c(C)nn(C)c2)=O)Cc2ccccc2C(CNC(C2CC2C(C)O)=O)C1 Cc1cccc(CC(=O)NC2CCCC(NC(c3cc(C)oc3C)=O)C2)c1 c1(NC(C(C)C)=O)ccc(N2CCN(C(c3ccnc(F)c3)=O)CC2)nc1 N1(C(COCC(=O)NC)=O)CC2CCC2(CCNC(c2cnc(C)cc2Cl)=O)C1 c1(CN=C(NC(COC)C)NCC(C)(C)C(C)(F)F)noc2c1CCCC2 CCCC(CNC(C1(C)CCC(O)CC1)=O)C(=O)NCC1CC(OC)C1 Cc1ccnc(C(=O)NCC2CCN(C(C3CC4C=CC3CC4)=O)CC2)c1O C(=O)(C1=C(C)S(=O)(=O)CC1)NCC1CCN(Cc2nc(CCCCC)[nH]n2)C1 N1(C(c2cc(Cl)cc(Cl)c2)C(=O)NCCCCCC)CC2(C)CCC2(C)C1 N1(C(Cc2cncc(C#N)c2)=O)C2CCC1C(F)C(NC(c1nsnc1O)=O)C2 C#CCCCCC(=O)NC1CCCC1CNC(c1cnoc1-c1ccoc1)=O Cc1c(C(N2CCC(C(=O)N(C)C(C)C)CC2)=O)ccc2c1OCCO2 N1(C(c2cnc(C)o2)=O)CCCC(CNC(c2cccc(C3CC3)c2C)=O)CC1 c1(OC)ccc(C=CC(=O)NCCC(C)NC(C2(C(C)C)CNC(=O)C2)=O)nc1 N1(C(=O)CCC2CCCCC2)CCCC12CCOC2=O.O=C1NN2CCCC12 c1(N(C(c2nnnn2CCOCC)C2CC(=C)C2)C)ccsc1OC.CNC c1(C(=O)NCCN(CCOC)Cc2cc(C)[nH]n2)ccc(C(N)=O)o1 C1(CCC)CCCCC1CSC.c12ccccc1C1CC1CNCc1cn-2nn1 C1(CNC(C(CC)NC(N)=O)=O)CCN(C(=O)CC2CCC(=O)N2)C1(C)C C1(N(C(=O)C(F)(F)F)C)C=CCN(CCC(=O)Nc2ccc(C(=O)CF)cc2)C1 C1(C(N2CCC(C)N(C(C3CC4CCC3O4)=O)CC2)=O)CCc2ccccc2C1 C(=O)(N=c1[nH]c(Cl)ncc1O)C1CCCN(C(c2c(C)nc(Cl)cc2Cl)=O)CC1 N1(C(=O)COCC2CCOC2)CCC2(CCN(C(c3cc4sccc4[nH]3)=O)C2)C1 C1(C(N2CC(OC)C(NC(=O)CNC(N)=O)C2)=O)CNC(=O)CC12CCC2 c1(CCNCc2c(OC)cccc2)c(Br)cncc1Br C1(OC)CN2CCCC2(C(N2CCOC(CNC(C3CC3(C)C)=O)C2)=O)C1 C1(C(=O)NC2CC3(CC(NC(CC)=O)C3)C2)CC(C)(C)SC(C)(C)C1 Cc1noc(C)c1CN1CC2C(C(=O)NCCCC3CCOCC3)C2C1 c1(C(N2C(C(C)(C)NC(c3cnns3)=O)CCC2)=O)cc2cc(Cl)ccn2n1 C1(CC(=O)NCC(CC)NC(c2[nH]cc(CC)c2)=O)CCCC2(CC2)C1 N1(C(C2(CCC)CCC2)=O)CC2CCC2(CCNC(=O)C(C)=CC(C)(C)C)C1 C1(CNC(C2CC3CCC2O3)=O)CN(C(c2ncc(C(F)(F)F)s2)=O)CCO1 C1(NC(C(C(CC)C)NC(c2cn(C)nc2OC)=O)=O)CC=C(C(C)C)CC1 CC(CNC(C1CN(C(N)=O)C1)=O)C(=O)N(C)CC1CCC1 CC1CCN(CC(=O)OCC2(O)CCC(C)C2)CC1 c1(C(=O)NC(C2CN(C(=O)C=Cc3ncc[nH]3)C2)C)ccc(-c2ccsc2)cc1 CC1(C)CCOC1CC(=O)NCC1CCCN1C(c1cnnn1C1CC1)=O C(=O)(CC1=NN(C)C(=O)C1)N1CC(OC)C(NC(C2CC(C)CC(C)(C)C2)=O)C1 c1(C(N2CC3C(NC(c4c(C)nc(O)cc4)=O)(C3)C2)=O)cccc2scnc12 c1(CNC(c2n(C)nc(C3CCCOC3)c2)=O)cc(Br)ccc1F c1(CC)cc(C(=O)NCc2ccc(CN(C(C)=O)C(C3CCC3)=O)cc2)n(C)n1 c1(COCC)nc(C(=O)NC(c2cncs2)C2CC2)c(-c2ccccc2)s1 c1(N(C)Cc2ccncc2)nnc(-c2ccc(Cl)nc2)n1CCC1CC1 N1(C(C(N2CCOCC2=O)C)=O)CC2CC(C1)CN(C(C1CCC(=O)N1)=O)C2 CC(C(=O)NCC(c1ccccc1)CNC(=O)CCC(=O)c1ccc[nH]1)C(F)F N1(C(CCSCC)=O)CC(NC(=O)Cn2cnc(C(N)=O)n2)C(C)(C)C1 C1(C(=O)OC)COCC(C)N1C(=O)NCCCCCOc1ccccc1 N1(C(C2CCC(C)O2)=O)CC(C)(C)CC1CNC(=O)CC1CCCOC1 N1(C(C(CC)C(C)O)=O)CCCC(C2CCN(C(C3CCC(F)CC3)=O)C2)C1 c1(Nc2ccc(CN(C)C(c3ccc(F)c(Cl)c3)=O)c(F)c2)c(Cl)cccc1Br N1(C(c2c(SC)scc2)=O)CC(NC(=O)Cc2ccon2)C(O)C1 C1(C(N2CC(n3cc(CNC(C4C=CCCC4)=O)nn3)C2)=O)CCS(=O)(=O)N1 c1(C(=O)NCC2C(NC(COCCOCC)=O)C2)cc(OC)c2occc2c1 CC1CCOCC1C(N1CCCC1(C)C(=O)NCCc1cscn1)=O c1(COC)ccc(C(=O)NC2CCCC2CNC(c2cnn(SC)c2)=O)cc1F N1(C(C)=O)CCC2(CC1)CC(NC(=O)CCNC(C)C)CCO2 c1(C(N2CC(NC(=O)Cc3csc(Cl)n3)C2)=O)cccc2c3c([nH]c12)CCCC3 C1(C(=O)NCC(=C)CCNC(c2csc(-c3ncccn3)n2)=O)CCC(=O)NC1 c1(C2CC2)nc2ncnc(N3CC(OC(=O)OC(C)(C)C)C3)c2s1.CC(C)S Cn1nnnc1SCCC(N1CCCC1CNC(=O)CSc1nncs1)=O c1(CC(N2CCCC(CC(=O)Nc3cncnc3Cl)C2)=O)ccc(O)c(O)c1 c1(C(=O)NC(C2CCN(C(=O)CS(=O)(=O)N(C)C)C2)C)csc2ncnc(O)c12 N1(C(=O)CCc2cccc(O)n2)CC2=C(C1)CN(C(C13CSCC1C3)=O)C2 C=CCC(F)(F)C(=O)NCC1CCCC1NC(c1sccc1-n1cnnn1)=O c1(NCCN(C(C2CCN(C)C(=O)C2)=O)CC)nnc2c(c1C(=O)OC)CCC2 C(C1=CCN(C(=O)CC2CCS(=O)(=O)CC2)CC1)NC(C1CCCS1)=O c1(C(=O)NC(CNC(C2(C)CCCCCC2)=O)(C)C2CC2)ccc2cnoc2c1 c1(C(=O)NCCCOCCNC(C(C2CCCOC2)OC)=O)nc(O)c(C)s1 CCC(C)CCC(=O)N(C1CN(C(c2cc(Br)oc2C)=O)CC1(C)C)C c1(C2C(C(N3CCC(NC(C4CC(O)C4)=O)CC3)=O)C2)ccc2c(c1)OCO2 N1(C(c2ncn(C)n2)=O)CCC2(CCCCN(C(=O)C(F)(F)c3ccco3)C2)C1 Cc1cnn(C)c1C(=O)N(C)CC1CCCN1C(C1CCCC2CC12)=O c1(NC(c2cccc(F)c2F)C(C)C)nc2c(s1)C(=O)NCC2 C1(C(=O)NC2CCCCC2NC(=O)COCc2nccn2C)(OC)CS(=O)(=O)C1 C1(C(N2CCCC(C(=O)NC3CC(C)(C(N)=O)C3)C2)=O)CCOC(=O)CC1 C=CCC(C(=O)N1CCCC1CC(=O)NCCc1cnn[nH]1)OC Cn1c(C(=O)NCC(C)(C)NC(C23CC(C(C)(C)C)(C2)C3)=O)cnc1S c1(CC(=O)N(CCNC(CC=C)=O)C)sccc1NC(=O)OCCOC n1(CC)nc(C(N2CCC(C(C)(C)NC(=O)CC3CCCCC3O)C2)=O)cc1O C1(C(=O)NCC2(CCC)CC2)CCCCC1(C)NC(c1cnc[nH]c1=N)=O Nc1cncc(C(=O)NCC(C2CCCCC2)NC(c2csnc2Br)=O)c1 c1(CC(N2C(CCNC(C=NOC)=O)COCC2)=O)cn2ccccc2n1 CC(C)C(O)C(C)C(=O)NCC1(F)CCCN(C(c2ccc(CO)nc2)=O)C1 CCCC(C(=O)N(CCCCNC(=O)Cc1ccnn1C1CCC1)C)N(C)C c1(OC)ccnc(N2CC(O)(C(C)NC(=O)CC3(CSC)CC3)C2)n1 N1(C(C2(COC)CCCO2)=O)CC2CC(NC(c3ccc(NC(C)C)s3)=O)C2C1 N1(C(CCOC)=O)CCCC(n2cc(CNC(c3ccc(C)o3)=O)nn2)C1 C1(CCOC)(NC(c2cnc(O)s2)=O)CCN(C(=O)Cc2cc(C)on2)C1 C1(NC(c2c(CCNC(C(C)OC(C)=O)=O)n[nH]c2)=O)CCCCCC1(C)C CN1CCC(C)(CNC(=O)C(C2CCN(C(c3ccc(CO)s3)=O)C2)F)C1 c1(C(N(C2CCN(C(=O)C(CC)NC(N)=O)C2)CCC)=O)scc(C)c1C C(=O)(CC(C)C(F)(F)F)NCC1(C)CCN(C(CC(C(C)C)O)=O)CC1 CN1CCOc2cc(CN3CC(NC(c4cc(F)cc(F)c4F)=O)C3)ccc21 Cc1nc(C(C)C)sc1C(N1CCOC(CCNC(=O)CC2COCC2O)C1)=O C(=O)(CC(C(=C)C)OCC)OCC.C=CC1CCC12c1nc(no1)COC2 N1(C(CCC(CC)OC)=O)CC2CC1CCN2C(c1cnn(CC)c1)=O c1(C(N2C(CC)C(NC(=O)C(C)OC(C)(C)C)CCC2)=O)cc2n(c1)CCCC2 c1(C(N(C2CCN(C(=O)CNC(N)=O)CC2)CCOC)=O)ccc2c(n1)CCO2 C12(NC(N3CC(c4ccc(Cl)nc4)(O)C3)=O)CCC1CCCN2 c1(C(N(C2CCC(NC(c3c(N)cnn3C)=O)CC2)C)=O)cc2sccc2[nH]1 C(=O)(C(=O)NC(C1CCCC1)CNC(C1CC1(F)Cl)=O)NCCOCC CCCC(CCC)CC(=O)NC(C)(CNC(=O)C(C)OCC)CC C1(NC(c2ncsc2Br)=O)Cc2ccccc2C1NC(C1CCC1)=O c1(C(=O)NCCCCN(C(CC(C)N(C)C)=O)C)ccc(=O)n(CCO)c1 c1(NC(C2C(C(=O)Nc3c(Br)ccnc3Cl)C2)=O)cc(Cl)ccc1[N+](=O)[O-] c1(N2CCC(CNC(c3c(OC)noc3C)=O)CC2)ccc(C)cc1[N+](=O)[O-] C1(CCNC(c2cnc(N3CCOCC3)nc2)=O)CC2CCC1C2 C1(C(C(=O)NCCC#N)N(C2CCCCC2(C)C)C)CCC2COCCC2C1 CC1(NC(C23CC2CNC3=O)=O)CCCCC1C(N1CC(C(N)=O)C2(CC2)C1)=O C(=O)(C1=NNC(=O)CC1)NCC(CNC(C1Cc2cc(C)ccc2O1)=O)OC C1(NC(CCOCC)=O)CCC2(CCC2)C1NC(=O)NCCOC(C)(C)C C1(CN(C)C(C2CCC(C(F)F)CC2)=O)CCN(C(c2cc[nH]c2)=O)CC1 C(c1c(C)nn(C)c1Cl)=CC(N1CC(CCNC(C2N(CC)C(=O)CC2)=O)C1)=O C1(=CCNC(C(c2cccc(Cl)c2)C)=O)CCN(C(C2(F)CC=CC2)=O)CC1 Cc1c(C(=O)NCCC(C)NC(c2cccc(C(F)F)c2)=O)nn(C)c1Br Cc1cc(NC(=O)COC(=O)C(C)Cc2cccc(F)c2)c(C)n1C(C)C C(=O)(C1CC(C)(C)Oc2ccccc21)N1CC(C(=O)NC2(C#C)CC2)OCC1 N1(C(C(CC)n2cccn2)=O)CC(CO)C2(C1)CN(C(c1ccoc1Cl)=O)C2 c1(C(CC)CC)nnc(N2CCOC(c3ccsc3)C2)n1CC(C)C N1(C(c2cn(CC)nn2)=O)CC2CCC1C(NC(=O)CNC(C)=O)C2 c1(C(=O)NC2CCC(NC(C3CCCC(C)(C)O3)=O)CC2)cnc2nccn2c1 N1(C(C(C)N(C)C)=O)CCCC12CCCN(C(C1CC(C(F)(F)F)C1)=O)C2 c1(CNCC(C#C)C2CCCO2)cc(COC)[nH]n1 N1(C(C2C(=C)C2)=O)CCC(C2CC2)C1CNC(=O)C(c1cccc(F)c1)C C(N=c1[nH]c(C2CC2(F)F)cs1)c1cc(C(=O)OC)no1 C=CC(CCC)CC(=O)NC(CCC)C(=O)NCCC(=O)N(C)C Cc1ccc2[nH]c(C(=O)NC3CC4CCC3N4C(c3ccn(C)n3)=O)cc2c1C CC1(C)CCC(C(=O)NC(C(F)(F)F)C2CC2)CN1C(c1c[nH]c(=O)cn1)=O N1(C(C(C)OC2CCCC2)=O)CC(CNC(=O)CCOCC(F)F)C(O)C1 C1(C(N(CC#CC)C)=O)CC2CC1CN(C(c1coc(C)n1)=O)C2 N1(C(C(=O)N(C)C)=O)C(C(=O)NC2Cc3ccccc3N2)C2CC(F)C1C2 c1(CN(C(c2[nH]cc(CC)n2)=O)CCN(C)C)c(C)nn(C)c1C C1(NC(C(C2(O)CN(C(CC3CCC(C)O3)=O)C2)F)=O)CC(C)(C)C12CC2 C(C(C)(C(=O)NCCSC(F)F)NC(c1ccncc1N)=O)SC C1(O)(CCNC(c2cncc(CC)c2)=O)CCN(C(=O)Cn2cnc(=N)[nH]2)CC1 C1(CNCc2cncc(Br)n2)CN2CCC1CC2 C1(CC(=O)NC2CC(CCNC(c3cnc(Cl)s3)=O)C2)CCS(=O)(=O)CC1 c1(C(=O)NC2CC(NC(C(CC)(C)COC)=O)C2)cc2cc(C)cc(C)c2[nH]1 CP(C)(=O)CN1CC(C(N2CCCC(NC(=O)CCc3nccs3)CCC2)=O)C1 C(=O)(N=c1[nH]nc(-c2cscn2)s1)N1CC(C)OC(C(N)=O)C1 C1(CC#C)(C(=O)N(C2CCCC2C#N)C)CCN(C(=O)Cc2cnc(C)s2)C1 CC(C)(C)CCC(=O)NCC1CCC1NC(=O)COCc1ccccc1Cl c1(C(=O)OCC)cnc(C)[nH]c1=NCC=CCNC(=O)C(C)S(N)(=O)=O c1(OC)ccc(Br)cc1C(N1CCC(C)(CNC(=O)C(O)CSC)C1)=O c1(CC(=O)N(CC(=O)N(C(C)C(=O)NCCC)C)CC#C)cc(C)no1 c1(C(N2CCN(C(=O)C3=CCCCC3)C3CCCC23)=O)cc(O)c2sccc2c1 CC1CC(NC(=O)Cc2cnccn2)CCN1C(c1ccc(F)nc1F)=O c1(C(N2CCCN(CCC#N)CC2)C(=O)NCC=C)ccnc(F)c1OC c1(CCC(=O)NCC(C)(C)OCCNC(C(C)C2CCC2)=O)nnc(C2CC2)o1 c1(OCC)ccc(C)nc1C(N1CC(C(C)NC(=O)Cc2ccc(Cl)nc2)C1)=O c1(C(C(=O)Nc2cn(C(C)C)nc2)C)cccnc1C(=O)NC(=O)CC(C)(C)C C1(O)(CNC(CNC(CCC)=O)=O)CCN(C(C2(c3ccno3)CCC2)=O)C1 Cc1c(F)cc(-c2cnc(C(F)(F)F)cc2C(=O)NCC2(C)CC2)cc1F N1(CC(=O)NC2CCCOC2)CCN(C(=O)C(n2nccc2C)C)CC1.CSC c1(C(=O)Nc2n(C)nc(Cl)c2)c(NC(C2CCCO2)=O)sc2c1CCCC2 C1(C)(C(=O)NCCC(C)NC(c2ccc(OC)c(Cl)n2)=O)CC(C2CC2)=NO1 C1(CNC(c2ncc(C)nc2)=O)CC2CCC1N2C(=O)CC1CCC(O)C1 C1(C(=O)Nc2c(OC)ncnc2)CCN(C(c2ccc(F)s2)=O)CC1O C1(OC)CN(C(C2CCC(=O)N2C)=O)CC1NC(c1conc1C)=O N1(C(C(C)(C)OCC)=O)CC(N(C(=O)CSc2ccc(F)cc2)C)C2(CC2)C1 C1(C(N(CCC)CCNC(=O)C(C2CCOCC2)O)=O)CCOC(C(C)C)C1 N1(C(=O)NCCCC(c2ccccc2)N(C)C)CCC(COC2CC2)C(F)(F)C1 c1(OC)ccccc1C(C)C(=O)NCCCCNC(c1sccc1Cl)=O Cc1c(C=CC(=O)NCCC(O)CNC(c2cc(F)cc(Cl)c2)=O)cnn1C C1(C2CC2)(CNC(c2cn(CC=C)nn2)=O)CCN(C(=O)Cn2ccsc2=N)C1 N1(C(C=CCCC)=O)CC(C)(C)CC1CNC(=O)C(C)SCc1ccccn1 c1(C(=O)NC2CCCC2NC(C2CC3CC(=O)C2C3)=O)cc2ccc(Cl)cc2[nH]1 c1(OC)ccc(C(N2CC(F)(CNC(=O)C(C)CSC)C2)=O)c2ccncc12 C1(CNC(c2cc(OC)no2)=O)CC(C(=O)N2CCCCC2C(C)(C)C)=NO1 c1(NCC2(C)CC(C)(C)C2)ccc(S(=O)(=O)N2CCCC(C3CC3)C2)c(Br)c1 N1(C(C=C(C)C)=O)CCC2CC12C(=O)NC(c1nc(=O)o[nH]1)C c1(C(=O)NCC(CO)NC(C(CC)NC(N)=O)=O)ccc(C(F)(F)F)cc1SC N1(C(c2cnn(C)n2)=O)CCC2(CC1)CC2(CO)CNC(=O)C1=CCCOCC1 C(C)(C(C(C)C)NC(=O)CC1CC(F)(F)C1)NC(C=CCOCCOC)=O N1(C(c2[nH]cc(CC)c2)=O)CCC2CN(C(=O)CSC(C)C)CCC12 C1(C(=O)NCCCCCN(C(C=C(COC)C)=O)C)CCCC(CF)C1 N1(C(C2(C)CCCC2)=O)CC2CC(NC(c3cnn(C(F)(F)F)c3)=O)CC2C1 C1(NC(CC(C)SC)=O)CC(NC(=O)C(C)N2CCCC2)CC1O c1(C(=O)NC(C)CNC(=O)Cc2ccoc2)cncn1-c1cnn(C)c1 C1(CNC(c2n(CCC)ccc2)=O)CN(C(=O)C=Cc2cnc[nH]2)CC1O C1(C(C)(C)NCc2cc(Cl)cc(Br)c2)CCc2ccccc2O1 CCCCC(O)C(=O)N1CCOC(CCNC(=O)CC(C)(C)SC)C1 c1(CC(=O)NCC(C2CCCC2)NC(=O)C=CC2CCCO2)csc2nccn12 C(=O)(CC1=CCN(C)CC1)NCCCC(C)NC(=O)C(F)CC1CCCC1 Cc1cccc(C)c1NC(=O)C(=O)NC(CN1CCCS1(=O)=O)C1CC1 c1(OC)nc(C(=O)NC(C)(CNC(C2CC2F)=O)C2CC2)sc1C C1(NC(C(C)N(C(C)=O)C)=O)(CNC(=O)C(C)(C)c2cccnc2)CCOCC1 c12ccc(cn1)CCSCCOCCNC(=O)C(=O)N2.c1(OC(N)=O)ccccc1 C1(C(=O)NCCC2CC(F)C2)(CC)CCCN1C(c1cc(CCO)on1)=O c1(C(N2CC3C(C2)N3C(c2ccc(I)cc2Cl)=O)=O)ccc(F)c(F)c1F N1(C(CC(=O)OC)=O)Cc2ccccc2C1C(=O)N1CCN(C)C(=O)C1C C(=O)(C1Cc2ccccc21)N1CC(NC(c2c(C)onc2O)=O)CC12CCC2 C(=O)(CC(C)(C)CSC)N1CC=CC(NC(C(C2CC2)SC)=O)C1 c1(NC(c2cnc(OC(C)C)c(Cl)c2)=O)ccc2c(n1)CCCN2 C12CC13CCN(CC3)C2=O.c1(C(=O)NCC2(CF)CC2)cn(C2CC2)nn1 Cc1cc(Cl)c(C(N2CC(NC(c3ccnn3C)=O)CC(O)C2)=O)cn1 C1(NC(Cn2nc(C)c(Cl)c2)=O)COC2(C1)CN(C(C1(O)CCCC1)=O)C2 c1(C(=O)NCC(CC)(C)NC(=O)C(C)S(N)(=O)=O)cnc2cc(C)nn2c1 n1(CCC(=O)NCC(C2CCC2)NC(C(C)N(C(C)=O)C)=O)c(C)csc1=O Cc1ccnc2c(C(=O)NC(CNC(=O)CN3CCCC3CO)CO)cccc12 C(=O)(C1CCCc2cccnc21)N(C(CNC(C1OCCO1)=O)C1CC1)C c1(CC(C)C)nnc(NC(=O)CC2CCN(C(=O)COCCOCCO)C2)s1 C1(C(N2CC(C)C(C)(CNC(c3cnncc3O)=O)C2)=O)Cc2ccccc2O1 c1(C(N2C(C(C)NC(C3N(CCC)CCC3)=O)CCC2)=O)cccc(Cl)c1O c1(C(=O)NC2C(NC(=O)Cc3ccc(Cl)cc3)C2)ccc(O)cc1C(F)F O=C(C1=NOC2(CCC2)C1)NC1CCN(C(C23COCC2C3)=O)C12CC2 c1(OC)ccc(C(=O)NCC(C(C)C(C)C)NC(=O)CC(C)C)cc1OC N1(C(=O)CCC2CC2)CCCC(C2CN(C(C3(C4CCCO4)CCCO3)=O)C2)C1 N1(C(C2C(C)C2C)=O)CCN(C(=O)C(C2CCOCC2)F)CC2(CC2)C1 C(C1=NOC2CN(C(c3ccnc(C)c3O)=O)CC12)NC(c1c(OC)csc1)=O CCC(C)(C(=O)N1CC(O)(CCNC(=O)CNC(=O)CN(C)C)C1)C(F)F CCC(c1ccc(C)cc1)=CC(N1CC(N(C)C)C(O)C1)=O C1(NC(C2CC3CC3C2)=O)COCCN(C(C2(C(F)(F)F)CCC2)=O)C1 C1(C(C)C)CCc2sc(C(N3CC4(CCC4NC(=O)C(C)C)C3)=O)cc2C1 C1(CC#N)(CC)CCCN(C(=O)NC2CC(=O)N(OCc3ccccc3)C2)C1 C1(NC(CCSC)=O)C(C)CN(C(c2cncc(OC3CCC3)c2)=O)CC1C N1(C(C(C=C)(C)O)=O)CC2(C1)CN(C(=O)CNC=O)CCO2 C(C)(C(CC(=O)N1CC(OC(F)F)C1)NC(C1(CO)CC(C)(C)C1)=O)OC C(=O)(C(C)(C)C1CCCN1C(C)=O)NC(c1ncc(C)[nH]1)CC.n12cc(nn1)C2 CC1(C)C(CNC(C2(SC)CC2)=O)CCN1C(C1CCCCN1C(N)=O)=O C12(NC(c3c(C)cn(C)n3)=O)COC(C1)C(NC(c1cc(Cl)cs1)=O)C2 N1(NCC(COc2cccc(C(C)C)c2)O)C(=O)NC2(CCCSC2)C1=O c1(CC(=O)NC2C(NC(CC(CCC)(C)C)=O)CCC2)ccc(S(C)(=O)=O)cc1 c1(C(=O)OCC)c(C)[nH]c(CN2CCC(NC(C3CCCO3)=O)C(O)C2)c1C CCCCCCC(C)C(=O)NC(COCC)C(=O)N(C)CCSC N#Cc1ccc(NC(C2CCN2Cc2ccccc2Br)=O)c2cccnc12 Cc1ccc(OC(C)C(=O)NC(C)(CNC(=O)C=Cc2ccsc2)CO)cc1 c1(C(N2CC(CNC(c3nc(Br)c[nH]3)=O)OCC2)=O)cn2ccnc2s1 C1(NC(C2(C)CCC(=O)NC2)=O)CC2CC(C1)N(c1cc(C(N)=O)ncn1)C2 C1(CC(=O)NCCC2N(C)CCC2)CC2(CC2)CN1C(C1CC2(CCO1)CC2)=O N1(C(C(CC)O)=O)CCN(C(c2cnn3cccnc23)=O)C2CCCC12 N1(C(Cc2ccc(C)s2)=O)CCOC2CN(C(=O)C(O)CCC(C)C)CC12 CCC(C)C(O)C(=O)N1CCC(CNC(=O)C(CCO)N(C)C)C12CC2 C12(C(=O)NC3CCC(N(C(CC=CCC)=O)C)C3)C(=O)C3CCC1C2C3 C#CC1(C(=O)NCC2=NOC(C)C2)CCN(C(=O)C(C)COC)C1 N1(C(c2cc(COC)on2)=O)CCC(CNC(c2cccc(OC)n2)=O)CC1C c1(-c2nn(C(C=C)C)c(-c3ccnn3CCOC)n2)ccc(F)c(Cl)c1 CC#CC1CCN(C(=O)CC2(CC(=O)OC)CCOCC2)CC1 Cc1c(NCC(C)CO)ncnc1N1CCC(C(N)=O)C1 N1(C(c2csc(C)c2C)=O)CC(C)(C(N2CC(S(C)=O)C2)=O)CC1(C)C c1(OC)ccc2nc(C(=O)OC(C(C)C)c3ncon3)sc2c1 c1(CNC(CCN(C(C(C)(C)c2ccno2)=O)CCCO)=O)cccc(C2CC2)c1 c1(C(=O)NCC2C(NC(c3cc(C)c(Cl)cc3F)=O)C2)cccc([N+](=O)[O-])c1Cl N1(C(c2ccc(CCC)[nH]2)=O)CCOC2(CCN(C(=O)CS(=O)(=O)C3CC3)C2)C1 C(=O)(C(F)C(C)C(F)(F)F)N1CCCC(CN(c2cc(SC)nc(SC)n2)C)C1 n1(CC(C)O)cc(C(=O)NCCCCCNC(c2ccc[n+]([O-])c2)=O)ccc1=O S(=O)(=O)(CCC(=O)N1CC2(NC(=O)CC3CCC(F)(F)CC3)CC1C2)N(C)C C1(CNC(c2cc(C)[nH]n2)=O)CC(NC(c2cnc(S)nc2)=O)C1(C)C N#Cc1ccc2c(c1)CC(CSCC(N1CC(N)C3CCCC3C1)=O)CO2 CCCC1c2ccccc2CCN1c1nc(Cl)nc2c1COCC2 Cc1cnc(NCc2cn(-c3ccccc3)nn2)c(S(=O)(=O)N2CC(C)CC2C)c1 C1(NC(C(CN(C)C)O)=O)COC2(C1)CN(C(c1csc(=N)[nH]1)=O)C2 C1(CC)CCCN(NC(=O)CCn2cc(COc3nonc3C(=O)O)nn2)C1 CCCCCCCCN(C(=O)CCC1CCCCN1C(c1ccsc1OC)=O)C N1(C(C2(C(C)(F)F)CC2)=O)CC2CC(C1)N(C(=O)CC(N1CCCCCC1)=O)C2 CN=c1nc(C(N2CCC(NC(=O)CC3CCC(=O)NC3)C(F)C2)=O)cc(C)[nH]1 N1(C(COCC)=O)CCc2sccc2C1CNC(c1ccc(Cl)c([N+](=O)[O-])c1)=O CC(C)CCCCC(=O)N(C1CN(C(=O)CCc2ccon2)CC12CC2)C N1(C(CCNC(=O)NC)=O)CCC(C(C(C)C)NC(=O)COC)CC1 CCC(C)(C)C(C)CC(=O)NC(C)C(CO)NC(c1cc(=O)c(OC)c[nH]1)=O c1(C(N2C3CN(Cc4cccc(Cl)c4)CC23)=O)ccc2c(c1)CCO2 Cc1ccncc1C(C)NC(C1CCCCN1C(c1cc(C2CC2)no1)=O)=O Cc1cccc2c(=O)c(C(=O)NC3CCN(C(=O)C(N)=O)CC3F)c[nH]c12 C1(CNc2nccc(OC)n2)CCCCN(C(=O)Cn2cnnn2)C1 c1(C(N2CC(NC(C3N(C(C)=O)CCOC3)=O)C(C)C2)=O)c(N)cc(Cl)cc1Cl N(C1c2ccccc2OCC1CO)C(c1cnc(C(C)C)s1)=O c1(C(=O)NCc2ccc(CCNC(C(CCC)C)=O)cc2)scc2c1OCCO2 c1(SC)cc(C(=O)NC2CCCC2NC(c2ccc(N)c(N)n2)=O)cc(Cl)c1 N1(C(C2C(C)(C)C2(C)C)=O)CC(NC(=O)CCCNC(=O)C2CC2)CC(O)C1 C1(C(=O)NC(C)C(F)(F)F)(COC)C=CCN1C(c1nc(Cl)cs1)=O C(=O)(CCC(=O)NCCCCN(C)C(C1CCCN(C(N)=O)C1)=O)OC N1(C(C(C)S)=O)CCOC(CC(=O)NCC2CC(=O)N(c3ccccc3)C2)C1 C1(C(N2C(C)CN(C(=O)C(F)(F)C3CC3)CCC2)=O)COc2cc(F)ccc2C1 c1(C(=O)NC2CCN(CC)C2)ccc(-c2ccccc2CNC)cc1 c1(C(=O)NCC(CC(=O)NC(c2cccnc2)CC)O)ccc(O)nc1C c1(C(=O)Oc2cccc(F)c2)cc(Cl)ncc1F.O=C1CCN1C1CNC1 C(=O)(C(F)CC(C)(C)C)NCC1(O)CCN(C(C2C(C(=O)OC)C2(C)C)=O)C1 c1(C(=O)NC2CCC(N(C(=O)Cc3ccoc3)C)C2)cncc(C(N)=O)c1 C1(OC)CC2(CCC(C(=O)NCC=CCNC(C3(C)CNC(=O)C3)=O)CC2)C1 N1(C(C(N2CCCCC2)C)=O)C(C(N2CC(N3CCC(O)C3)C2)=O)CC1C C1(NC(C(CC=CC)C)=O)CC=C(C(=O)N(C2CC2)Cc2cnn(C)c2)C1 C=CCCCCCCC(=O)N1CCCC(C(=O)NC2COCC2F)C1C c1(C(N2CCC(COC)(CNC(=O)CN(C)C(C)=O)C2)=O)ccc(C)c(F)c1F Cc1sc2ccccc2c1C(=O)NCC(C)CN(C)C(C1(F)CCCCCC1)=O c1(N(C)C)cnc(C(=O)NCC2(O)CN(C(c3cnc(S)[nH]3)=O)C2)nc1 N1(C(C2C(C)(Br)C2)=O)CC2CCC1C1CN(c3nc(-c4ccccc4)ns3)CC21 N1(C(C(CCCOC)C)=O)CCCCC(CNC(c2ncoc2C)=O)CC1 n1(CCC)cc(CN(C(C(=O)NCc2cc(C)on2)C2CCOC2)C)c(C)n1 C1(C(C)C)CC(CC(=O)NCC(C)(C)CN(C(=O)Cc2cnn(C)c2)C)CCO1 Cc1cc(N2CC3C(C2)C3(C)C)nc(N(C)CC2CCCS2)n1 Cc1nccn1CCC(=O)NCCCOCCC(=O)NCC1CCSC1 c1(C(N2CC(C)(CNC(C3CNC(=O)N3)=O)OCC2)=O)cc(F)c(F)c(Cl)c1F Cc1nc(C(N2CCC(O)C2C(N2CCC(c3cnco3)C2)=O)=O)c(C)s1 C(=O)(CCCC(F)F)NCC(CC)NC(=O)C(C)n1ccnc1 C1(C)(CNc2c(C(N3CCC(C)CC3)=O)cccc2)CCS(=O)(=O)N1C C1(CNC(C(=Cc2ccco2)C)=O)CCCCC1NC(C1CC(=O)N1)=O C1(CC(=O)NCC(CC)N(C(=O)CC2CCC(=O)NC2)C)NC(=O)NC1=O C(=O)(C(CNC(C1(C(F)F)CC2(CC2)C1)=O)C(C)C)N(CCC(C)C)C1CC1 N1(C(c2cc(COC)on2)=O)CCC(NC(=O)Cc2ccc(C)cc2)C1C(C)C N1(C(C2CCCN(C(C(CN(C)C)O)=O)C2)=O)CC(C(N)=O)C2(CC2)C1 C1(NC(c2ccn(C(C)C)n2)=O)CC=CCC1C(=O)NCC1(O)CCCOC1 C(=O)(C(C)C(C)S(C)(=O)=O)NC12CC(NC(Cc3c(C(=O)OC)occ3)=O)(C1)C2 CC(CC(=O)NCC12CCC(NC(=O)C(C)n3cncn3)(CC1)CO2)C(C)(C)C N1(C(c2ccc(-c3nc(C)c(C)o3)cc2)C(=O)NC(C)C)CC(C)SC(C)C1 c1(CC)ccc(CC(=O)NC2CCCC2NC(=O)C(C)C(C)C)cc1F C12(NC(c3c(CC)cccn3)=O)CCN(C(c3[nH]c(C)nc3C)=O)CC1C2 c1(C(=O)NC(CC)CNC(=O)Cc2cc(C)ccc2C)n[nH]c2ccc(F)cc12 C(=O)(C1=C(C#N)CCC1)N1CC(CNC(Cc2cc(C)[nH]n2)=O)C(C(F)(F)F)C1 O=S(=O)(c1ccc(N2CCOC(c3ccccc3)C2)cc1)C(F)(F)F N1(C(=O)NC(c2nccc(C)c2)C)CC2(C1)CN(C)C2 c1(CC(=O)NC2CN(C(CC(=C)C)=O)C(C)CC2)c(C)[nH]c2ccccc12 CCC(O)CCN=c1nc(N2CCC3(CCN(S(C)(=O)=O)CC3)C2)cc[nH]1 N1(C(COC(C)C)=O)CC(O)CC1CO.C12CC(O)C1CC(=O)N2 C1(NC(c2onc(C)n2)=O)CN(C(C2CC(F)(CO)C2)=O)CC1C C1(NC(C=CC)=O)(CC)CCN(C(=O)C(C2CCC2)OC)CC1 NS(=O)(=O)CCC(=O)NCCC1CCC(NC(C2CC2C2CC2)=O)C1 C12(COC)CC(NC(=O)CC(C)CN(C)C)(CN1C(c1ccc(OC)s1)=O)C2 C1(=CCNC(C2(CCOC)CC2)=O)CCN(C(=O)C(=O)N(C)C)CC1 C1(CNC(C(C(C)C)(C)O)=O)CCC2(CN(C(=O)CCn3cncn3)C2)O1 c1(C(=O)NCC2(OC)CN(C(=O)C(F)(F)C3CC3)C2)cnc2nccn2c1 CC(C)C(C(=O)NC1CCC(OC(F)F)C1)N1CCCCC1c1ncc(Br)cn1 C1(NC(c2cc(C(F)(F)F)n[nH]2)=O)CCN(C(C2CCC=CCC2)=O)CC1O N1(C(c2c(CCC)n[nH]c2)=O)CCCCC1C(=O)NCC(C)N(C)C1CC1 c1(C(N2CCC(C(C)(C)NC(=O)C3=C(Cl)CC3)C2)=O)cc2c(cc1Cl)OCO2 C1(NC(C2(OCC)CCC2)=O)CC2CC(NC(c3ccoc3C(C)C)=O)C1C2 Cc1cc(C)c(C=CC(=O)NC2CC2CNC(=O)CC(C)(C)CC(F)F)c(C)c1 C(C1=CCN(C(c2ccn(C)c2C2CCC2)=O)CC1)NC(CCSCCCC)=O C1(OC(C(c2cccc(O)n2)C)=O)CCN(c2ccc(Cl)cc2)C1=O c1(C(=O)NCCCN(C(C2OCC(C)C2)=O)C)c(Cl)cnn1C(C)C C1(C(=O)NC(C)CCCNC(=O)COC2COC2)CNC(=O)CC12CCC2 CC1(C)CC(NC(c2ccc(C(C)(C)C)c(Cl)c2)=O)CN(C(c2csnn2)=O)C1 CC(N=c1[nH]c2c(c(=NCCC3CCCO3)[nH]1)CCC2)c1cccc(Cl)c1 C1(NC(C=C(C)C)=O)CCCC(CNC(=O)Cc2cscc2F)C1 CC1(C)CCC(CNC(c2sc(F)cc2Cl)=O)N(C(=O)COCC2CCC2)C1 Cc1cc(C)c2c(S(=O)(=O)NC(c3nn(C)c4ccc(Br)cc34)=O)n[nH]c2n1 C1(CC(C)C)CCCC1NC(C1(N(C)C(C2CCCSC2)=O)CC1)=O c1(C(N(C(C)CNC(=O)CN2CC(C)(C)C2)CC)=O)ccc(C2CC2)c(OC)c1 Cn1cnc(C(=O)NCCN2CCN(C(c3nc(Cl)ccc3N)=O)CC2)cc1=O C(=O)(CS(=O)(=O)C1CC1)N(CCn1cc(Cc2ccc(Br)cn2)nn1)CC N1(C(C(C)N(C(=O)C=CCN(C)C)CCC)=O)CCC(c2nn[nH]n2)C1 CC(C)C(CNC(=O)C=Cc1cnn(C)c1)C(=O)N(C1(C)CCCC1)C C(c1scnc1C)=CC(=O)NC1C(NC(C(C)(c2ccccc2)OC)=O)COC1 N1(C(CC2N(C)CCOC2)=O)CCC(O)(Cn2cc(C(C)(C)C)nn2)CC1 N1(C(CC(C)(C)C)=O)CCN(C(=O)CSc2ccccc2O)CC1c1cn[nH]c1 C1(C(=O)NCCN(CCOC)C(c2nnsc2SC)=O)CCC2(CCC2)C1 c1(OC(C(=O)NC2CC(N(C(C=C(CCC)C)=O)C)C2)C)ccccn1 c1(C(=O)NCC2CCN(C(CCc3cnc(C)o3)=O)C2)cnncc1C N1(c2snc(C)n2)CC(NC(C2CCC(F)(F)CC2)=O)CC2(CCC2)C1 Cc1ncccc1CNC(=O)COCC1CCCCN1C(=O)CC1(C)OCCO1 N1(C(C2C(C)C2)=O)CCC2(CC1)CC(NC(c1cc(Cl)cs1)=O)CO2 c1(NC(C2C3CN(Cc4cn(CCC)nc4)C2C3)=O)cc(O)cc(O)c1 c1(C(=O)NCC2C(C)CN(C(=O)C(F)(F)C(F)F)C2)c(O)nnc2c1CCC2 CCC(CC(C)C)C(=O)N1CCC(NC(=O)C(C)C(C)(F)F)C(CO)CC1 c1(CC)ccc(C(=O)NCCOCC(=O)NCCN(C(C)C)CC)cc1 C1(NC(C(Cn2ccnn2)NC(C2C=CCS2)=O)=O)CC2CCCC(C1)C2 CC1CCN(C(c2cc[nH]c(=N)c2)=O)CC1CNC(c1[nH]ccc1C1CC1)=O c1(CC)cc(C)c(C(=O)NC2(C(=O)NC3CCNC(=O)C3)CCOCC2)o1 c1(C(=O)NCC2(F)CN(C(c3c(C)con3)=O)C2)sc(C)c(C)c1C Cc1c(Cl)ccc2c(CC(=O)NC3CCC(NC(C4(C)CC4F)=O)CC3)coc12 C1(CC(=O)NCC(C)(C2CC2)NC(C2N(CC)CC2)=O)NC(=O)NC1=O C#CC1(NC(c2ccc(CNC(=O)C(CCC)N(C)C)s2)=O)CCCCCC1 C=CCCCCCCCCC(=O)NC(CNC(=O)C(C1CCCCCC1)C)CO S(=O)(=O)(c1ccc([N+](=O)[O-])cc1NC(N1CCC2OCCC2C1(C)C)=O)NC C1(C(=O)NCC2CN(C(c3n(CC)ccc3)=O)CC2C)CC(C2CC2)=NO1 C1(N=c2cc(Br)n(C)[nH]2)(c2n(CCSC)nnn2)CCC2CC12 CC(C)C(CNC(C1CCN(C)C1)=O)C(=O)NCC1CCCCO1 N1(C(CCc2n(C)cnc2)=O)CC=CC(NC(C2(C)CCCS2)=O)C1 C(C(O)CC(=O)N1CCC(OCCN(C)C)C1)NC(C(C)=C1CCCC1)=O C(=O)(CS(=O)(=O)CC)NC(CCNC(CC(CC)C)=O)Cc1ccccc1 Cc1ccc(NC(C2CCN(c3ncc4c(n3)CCC4)C2)=O)cc1[N+](=O)[O-] N1(C(c2c(CC)nns2)=O)CC(CCNC(C2(C3CC3)CCCO2)=O)OC(C)C1 c1(CC(N2CCC(NC(c3ccc(C)cc3Cl)=O)CC2)=O)csc2cc(C)sc12 n1(CC(N2CCC(F)(CNC(CC(CC)C)=O)C2)=O)cc([N+](=O)[O-])ccc1=O C(=O)(C(C)(C)C(C)(F)F)N1CC(CC(C(=O)NCC(C)(C)F)F)C1 c1(C(N(CCC2CCN(C(CCCSC)=O)CC2)C)=O)cc([N+](=O)[O-])cnc1O c1(C(N(CC(CN(C(C(C(C)(C)C)OC)=O)C)O)C)=O)c(F)ccc(C)c1Cl c1(CN(c2cc(NC(c3ccco3)C)ncn2)C)ncc(Cl)cc1F N1(C(CCC=CC)=O)CCCC2CCN(C(c3cn4ccnc4s3)=O)CC12 N1(C(c2cn(CC)nc2)=O)CCN(C(=O)C=C2CCN(C)C2)CC1CF c1(C(=O)NCC(CCC)C)cc(S(=O)(=O)CC)ccc1OC N1(C(c2nnn(C)n2)=O)CCC2CCCC12CNC(c1cnc(N)cn1)=O C(=O)(CC1CNc2ccccc21)N(CCOC)CCNC(=O)C=Cc1nccs1 N1(C(CC=CC=C)=O)CCc2ccccc2C(NC(=O)C=CCC)C1 N1(C(C(F)=C(C)C)=O)CC2CCC1C1CN(C(c3c(C)noc3N)=O)CC21 C1(NC(c2nnc(O)nc2O)=O)CN(C(=O)CCCn2ccnn2)CCC1CO C1(Oc2ccc(N(C(CSCC(=O)OC)=O)C)cc2)CCCN2CCCC12 Cc1ccc(C(=O)NC2CCC(CNC(C3CCC(N(C)C)C3)=O)C2)o1 C1(OC(C)(C)C)N(OCC(=O)NCC2CN(C(C(CC)C)=O)C2)CCC12CCC2 S(=O)(=O)(c1cccc(Br)c1)NC(C)C(N1C2CCC1CC2)=O N1(NC(=O)NCCC(=O)NC(C)CCN(C)C(C2CCCC2)=O)CCSCC1 C1(NC(=O)CCOC2CC2)COC2CN(C(=O)CC=CCc3ccccc3)CC12 C12(NC(=O)CC3CCCS(=O)(=O)C3)CCC(CN(C(=O)C3=CCCCC3)C1)C2 N1(C(C2C(COC)CC2)=O)CC=CC1C(N1CCC1)=O N1(C(c2ccn(C)c2)=O)CC(O)CCC1C(=O)NCc1cnn(C)c1O N1(C(CN(CCC)C)=O)CCCC(NC(c2coc(C(=O)OC)n2)=O)C1 O=C(N=c1[nH][nH]c2c1CCCC2)C1CCN1C(c1cccc(CCO)c1)=O CCC(CC)(CCC(=O)OCC)NC(c1nnnn1CCCF)C1CCC1 C(CN=c1nc(CO)[nH]s1)=C(CNC(C1CCC(C(C)(C)C)CC1)=O)CCCO N1(C(CCC#C)=O)CC(C2CCCN(C(C3CCCCN3N=O)=O)C2)C1 Cc1occc1CC(=O)NCC12CC(NC(c3ccn(C4CC4)n3)=O)(C1)C2 CN1CCCC1C=CC(=O)NCCC1CN(C(c2n[nH]cc2Br)=O)C1 N1(CC)CCN(CCCC(N2CCC(NC(=O)C(C)=C(C)C)C2C)=O)CC1 Cc1csc(CC(=O)NCC(C2CCCC2)NC(=O)Cc2csc(C)n2)c1 C1(CNC(COC2(C)CN(C(CSCC)=O)C2)=O)COCCN1CC N1(C(c2c(Br)cn(CC)n2)=O)CCC(CNC(C2CCOC2)=O)C(O)C1 C1(NC(CC)=O)CCCCC1NC(C1CC1OCc1ccccc1)=O C(=O)(CCCC(C)(C)NC(c1ccccc1OC)=O)NCC#C c1(OC)cc(C(=O)NC(CNC(C2(O)CCCCC2)=O)CC(F)(F)F)cc(F)n1 N1(C(c2n(CC#C)ccc2)=O)CCC2(CCCN(C(C3CC(F)(F)CS3)=O)C2)C1 c1(COC)cccc(C(=O)NC2CCC(CNC(=O)CCc3ncccn3)C2)c1 C1(C(=O)NCC(c2cccs2)C)CCN(C(C2CC2C(C)(F)F)=O)CCO1 C(=O)(C(CC)(CC)CC)N(C)CC1CCN(C(c2nc(CC)oc2C)=O)CC1 N1(C(c2c(C)coc2)=O)CCC2(CC2C(=O)NCc2cccnc2C)C1 c1(C(=O)NCCCNC(c2c(C)csn2)=O)c(C)nsc1C Cc1ccc(NC(=O)C(=O)NC2CN(C(=O)CS(N)(=O)=O)CC2O)cc1C CCC(C(=O)NCC12CC(NC(c3cn(C)nc3SC)=O)(C1)C2)C(C)(C)CC c1(CN(CCN(C(c2c(C)cn(C)n2)=O)C)C)nc2ncccn2n1 C(C(C)(C(=O)N(C)CC12CCC(CC1)C2)NC(=O)C(CN(C)C)N(C)C)SC Cc1nnccc1C(=O)NCCC1(NC(=O)COC2CCOC2)CCCC1 CCCCC(O)C(C)C(=O)N1CCC(C2CC2)C1C(=O)NCCC1(O)CCC1 CC1C(NC(=O)COC2CCOCC2)CC2CCC1N2C(C1CCN1C)=O c1(CCC(=O)NC2CC(NC(C(C=C)O)=O)C2)c(C)noc1C N1(C(C(CC)(C)O)=O)CC2(C(N3CC(O)C(N=[N+]=[N-])C3)=O)CCC1CC2 n1(CC(=O)NCC2CCC2C(N2CC(SC(F)F)C2)=O)cnoc1=O N1(C(Cn2c(=N)scc2)=O)CC2CC(NC(C3CCCN3N=O)=O)C2C1 C1(OCC=C)CCN(C(c2cnn(CC(F)F)n2)C(=O)NCCCC2CC2)CC1 c1(-n2cc(C(=O)NC3(C4CCCO4)CCC3)nn2)ccc(Cl)cc1Cl C(=O)(CC(O)(C(F)(F)F)c1nccn1C)NC(c1ccc(CC)cc1)CC(=O)O c1(C(=O)Nc2cc(C(=O)OC)ncc2)cccc(=O)n1C.C12(CC1)C(=O)NC2 c1(C(N(CC(O)CNC(=O)CSc2n[nH]c(O)n2)C)=O)cccc([N+](=O)[O-])c1Cl C(=O)(C(C(C)NC(c1coc(CO)c1)=O)C(C)C)NC(CC(=O)OCC)C N1(C(CC2C(C)CCO2)=O)CCN(c2ccc(NC(=O)COCCF)cn2)CC1 c1(C(=O)NC(CC)C(=O)OC)ccc2c(-c3cccc(OCCF)c3)n[nH]c2c1 c1(C(N(C2CCN(c3nc(O)c(C)s3)C2)CCC)=O)cc(O)nc(C)n1 C=CCCCCN(C(COC(C)(C)C)C(=O)Nc1ccccc1)C C(N=c1nc2scnc2c(NC2CC(C(C)(C)C)C2)[nH]1)c1ccn(C)n1 c1(C(=O)NCC(CO)NC(C2CN(c3nncs3)C2)=O)cc(F)c(O)c(F)c1 C=CC1(C(N2CC(OCC3CCN(C(=O)CC4CC4C)CC3)C2)=O)CCCCC1 N1(C(CCCN(C(C)=O)C)=O)CC2CC1CN2Cc1ncnn1C(C)(C)C N1(S(CCCC)(=O)=O)CC2CCN(C(C3CCCN3C(C)C)=O)CC2C1 C1(C(N2C(C(=O)NC(c3cc(C)on3)C)CC(C)C2)=O)CN(C)CC(C)O1 c1(NC(c2cccc(OCC)c2)c2nnnn2CCOC)cccc(C#N)c1C C1(CNC(=O)C(C2CCCCC2)F)(NC(C2CC2C2CCCO2)=O)CCOCC1 c1(C(N2CC(CNC(C3C(C=C(C)C)C3(C)C)=O)C2)=O)cc[nH]c(=N)c1[N+](=O)[O-] N1(C(c2c(CNC(C3C(C)(C)C(=O)C3)=O)c[nH]n2)=O)CC(O)CC1(C)CO Cc1c(C(=O)NC2(C)CN(C(=O)C(C(C)C)NC=O)C2)ccc(F)c1F C1(NC(c2cc(C(C)(F)F)n[nH]2)=O)C=CCN(C(=O)Cc2cn[nH]c2)C1 O(N1CCC(CC(=O)NC(C)C(C)NC(=O)Cc2noc(C)c2C#N)CC1)CC c1(OC)ccc(F)c(N)c1C(=O)NC1CC(C)(NC(=O)C=Cc2ccccc2)C1 CC1CN(C(C2CCC(O)CC2)=O)CCCN1C(c1cnnc(Cl)c1)=O c1(C(=O)NCCC(C)NC(C(C=CCCC)O)=O)cnc(N)c(O)c1 C(=O)(C(CCSC)NC(c1ccncc1F)=O)NC1CC(OCC)C1 c1(C(=O)OC)csc2cc(C(N3CC(NC(C4CC4CF)=O)C(C)C3)=O)sc12 c1(C(=O)NCCOCCCNC(C2CC2Cl)=O)ccc(SC(F)F)cn1 CC1CCC(CNC(c2cc(F)cnc2O)=O)N(C(=O)C2=CCOC2)C1 C1(CN(C(=O)NCc2c(OC)cnc(C(F)(F)F)c2)C)COc2ccccc2O1 C(C)(C(=O)NCC1CCC1C(=O)NCCCCOC)OCC.C1CC1 CCCC(CCC)CC(=O)N1C(CNC(=O)CC23CC(C2)C3)CC2CCCCC12 C1(c2cc(CNC(C=C(CCC)C)=O)on2)CCN(C(c2cncn2C)=O)CC1 CC1CC(NC(c2c[nH]ccc2=N)=O)CN1C(c1cc(C2CC2)oc1C1CC1)=O CC1CCC(C(=O)NC(c2csnn2)C)CN1C(=O)COCC1CC1 C(CC(C)(C)C(=O)NC(C)CCNC(c1cc(Br)sn1)=O)OC C1(C(=O)Nc2cncc(COC)c2)(C(=O)NCCN(C)CCO)CNC(=O)C1 Cc1oc(S(C)(=O)=O)cc1C(=O)NCC(C)(O)CNC(=O)C(C)(F)F C1(C(=O)Nc2cccc(NC(C3C(c4n(C)nnc4)C3)=O)c2)CCOCC1(C)C c1(C(C)OC)nc(Cl)cc(=NCC2CCC(NC(c3nc(Cl)cs3)=O)C2)[nH]1 C1(CC)C(C)CCN1C(c1ccc(C2CCCC(=O)N2)cc1)=O c1(C(=O)NCC2CC(NC(C3(CC)CCC3)=O)C2)oc(CO)cc1C C(=O)(C1CCc2c[nH]nc21)N1CCCC(CNC(c2c(CC)onc2)=O)CC1 c1(C(N2CC(N3CCN(C(C4(CC=C)CC4)=O)CC3)C2)=O)ccn2ccnc2c1 C(=O)(C(CC(F)F)NC(=O)CN1CSCC1=O)NCC(C)CCO Cc1nc(N2CCCC2C(=O)Nc2ccc(N(C)C)cc2)sc1F Cc1c(CC(N2CCCC(CNC(c3cc(Cl)no3)=O)C2)=O)sc2ccccc12 CCC(C)C(O)CC(=O)NCc1n[nH]cc1C(=O)NC1CCS(=O)CC1 N1(C(C2(C)CC(=O)C2)=O)CCN(C(C2(C#N)CC3CC3C2)=O)CC(O)C1 S(=O)(=O)(c1cccc(=NCCOc2ccccc2)[nH]1)N(C1CC1(C)C)C c1(OC)cc(C(=O)NC(C)(CNC(=O)CC(C)NC(N)=O)CO)cc(OC)c1C N1(C(c2cc(OCC)n[nH]2)=O)CCC2CN(C(=O)CN3C(=O)CCCC3=O)C2C1 C=CC(CC)C(=O)NCC1(CNC(c2cnn(C(C)(C)C)c2)=O)CC12CCC2 C1(NC(C2(N3CCN(C)CC3)CC2)=O)CN(C(=O)CC2CCC2)CC2(CC2)C1 N1(C(c2c(C)cccc2F)=O)CC2CC(C1)N(C(=O)CN1C(=O)CNC1=O)C2 CC1(O)CCC(CC(=O)NCC2CC(NC(=O)C(F)CC3CC3)C2)CC1 C(=O)(CC(F)(F)C(F)(F)F)NCC1(OC)CN(C(C23CCC(CC2)C(C)O3)=O)C1 N1(C(CCC(C)SC)=O)CCCCCC1C(=O)NCCC1CCC(=O)N1 C1(C(=O)NC2(CNC(c3c(C)oc(C(F)(F)F)n3)=O)CC2)CCc2ncnn2C1 CC(C)CCCC(=O)NC1CC2C(C(=O)NCC3CCCCCN3C)C2C1 S(=O)(=O)(C1CC2(CC2)C1)N1CCCC(C(N2CCCC(C(N)=O)C2)=O)C1 N1(C(CCCC=C)=O)CCN(C(=O)Cc2ccc(F)cc2C)C(C)C1C CCC(CC(=O)NCC1CC1NC(=O)C(F)(F)c1csc(C)c1)C1CC1 C(CC)(CCC(=O)NCC(C)(C)C#N)NC(COCCC)=O c1(CC)ccc(C(=O)N(C)CC2CCN(C(=O)Cc3ccc(C)o3)C2)cc1F c1(CC(=O)NC2C=CC(CC(=O)NC(CC=C)CC=C)C2)cccc(C#N)c1 c1(C(N(C(CC)CC(=O)OCCCC(=O)N(C)C)C)=O)cc2cccnc2[nH]1 c1(CC(=O)NC(CN(C(CCN(CC)CC)=O)C)(C)C)coc(C(F)F)n1 Cc1cc(C(=O)NCCc2ocnc2CNC(c2[nH]c(C)nc2C)=O)c(N)c(C)c1 C1(NC(C(C(C)C)O)=O)CCC(C)N(C(C2CCC(=O)N(C3CC3)C2)=O)C1 Cc1nn(-c2ccncc2)cc1CN(CC(O)C(C)(C)C)C C1(O)(C(=O)OC)CN(C(CCC2CC2)C(=O)NC(C)C)CC1O CCC(C(=O)NOCC(=O)NC1CN(CC)CC1C)N(C)C C1(NC(c2nccc(OC)c2)=O)CN(C(=O)C(C)NC=O)CC12CC2 N1(C(c2c(OC)csc2)=O)CC(CNC(=O)CC(C)CF)C2(CCOCC2)C1 N1(C(CC(C)SC)=O)CCN(CCCCCNC(=O)Cc2cc[nH]c(=N)c2)CC1 N1(C(CC(C)F)=O)C2CC1CN(C(c1ncc[nH]1)=O)C2 c1(CS(=O)(=O)Oc2ccc(CF)cc2)cc(F)c(F)cc1Cl C(C(=O)NCC1CCCCCC1)(C(C)C)CC.C12CCN(CC1)C2=O CC1(C)CC(CNC(c2ccccc2Cl)c2nnnn2CCC2CC2)CNC1=O C12(CNC(C(C)(C)F)=O)CCC(CC1NC(C1CC1c1cc(F)ccc1F)=O)C2 CCC(C)C(=O)C(=O)NCC1(O)CCN(C(c2cc(C)sn2)=O)CC1 C1(C2CC2)(CNC(c2n(C=C)ncc2)=O)CCN(C(c2cc(C)ncc2C)=O)C1 N1(C(CCN(C(C)=O)CCO)=O)CCC(F)(CO)C1 c1(C(=O)NC(C2(O)CN(C(C3CC(OC)C3)=O)C2)C)sc(Cl)cc1Cl C1(NC(C2CC2F)=O)CCN(C(=O)CCc2csnn2)C12CCC2 N1(C(C(CC(C)C)NC(c2cc(C)nn2C)=O)=O)CCC(C)(C2CC2)C1 Cc1ccc(C(N2CC(N3CCN(S(=O)(=O)CC4CCC4)CC3)C2)=O)c(F)c1 CCC(CC(=O)NC(c1ccsc1)C)NC(=O)Cc1csnc1C C1(NC(CC2CCN(C(CCC=C)=O)CC2)=O)CCOC12CCOC2 N1(C(CN(C)C(N)=O)=O)CCC(C2CCN(C(c3cc(C4CC4)ccn3)=O)C2)C1 c1(C(=O)NC(c2cccnc2)C(=O)NCCC(C)OC)c[nH]ccc1=O C12(NC(=O)CCF)CCCN(CC(F)(F)F)CC1C2.c12cccc(n1)NC2=O c1(C(N(CC(C)N(C)C(c2nnn3c2CSCC3)=O)C)=O)csc2c1CCCC2 c1(OC)nc(-c2occc2C)ccc1C(=O)NCCC#N N1(C(CCC)=O)CCCC12CCN(C(=O)C(C(C)C)n1cc(Br)cn1)C2 C1(C(=O)NC(C)CC(F)(F)F)CCN(C(C2CCCCC(=O)N2)=O)C(C)(C)C1 N1(C(CC2ON=C(C)C2)=O)CCC(N(C(=O)CC2(O)CCOCC2)CCO)CC1 N1(C(CC2CN(C(C)=O)C2)=O)CCC2CCCC12CNC(=O)C(C)c1ccco1 c1(C(=O)NC(CN(C(C(C)C2CCCC2)=O)C)(C)C)ccc2c(c1)nnn2C c1(C(=O)NCC(CC(C)C)NC(C2(C)CC2C)=O)cnc(N)c(Cl)c1 C(=O)(C1=NNC(=O)CC1)NC1C(C)CN(C(c2sccc2C(F)F)=O)C1 c1(CC)cc(NC2CN(C(c3n[nH]cc3C)=O)CC2C)nc(C)n1 CCC(C)(CCNC(=O)Cc1ccc(O)nc1)NC(=O)C(=Cc1cccnc1)F c1(CC)ccc(NC(C2CC(OC)CN2C(=O)CN2CCCCC2=O)=O)cc1 Cc1cc(Cl)cc(N)c1C(N1CCC(C(C)(C)C)C1)=O CC(C)C(C)CC(=O)NC1(CNC(c2ccc(Cl)cc2Cl)=O)CCOC1 c1(NC(=O)NC2(C(=O)OC)CCC3(CC2)CC3)cnc2ncccc2c1 C1(F)(CNC(c2n(C(C)C)ccn2)=O)CCN(C(C2CCC(C)(F)CC2)=O)CC1 c1(CCNC(=O)NC(CC(=O)OCC)C2CCCCC2)c(F)cncc1F c1(C(=O)NCC(CCNC(C(C)CC(N)=O)=O)(C)C)cccc(S(N)(=O)=O)c1 N1(C(c2c(C)nc(O)cc2)=O)CCC(C)(C)C(C(N2CCN(C)C(=O)C2)=O)C1 Cc1occc1C(N1CCCC1CCNC(C1CC1(C)C(F)F)=O)=O S(=O)(=O)(c1ncc[nH]1)Nc1scc(C(=O)NC2CC=CCC2)n1 C1(NC(C2CCCN(C(CC3CCCC(C)(C)C3)=O)C2)=O)CN2CCC1(C)CC2 C(=O)(C#CC1CCCCC1)N(C1CCCCN(C(C2N(C)CCC2)=O)C1)CCO c1(CN2CC3C(CN(CCOC)C)C3C2)cc2c[nH]nc2cc1C Cc1ccnc(C(=O)N(C)CC2CN(C(=O)C(n3ccnc3C)C)CCO2)n1 c1(C(=O)OCC)cc(C)ccc1S(=O)(=O)Oc1cccc(N(C(C)C(C)C)C)c1 N1(C(Cc2cccc(C)c2)=O)CC2(CCCC2NC(C2CC3CCC2C3)=O)C1 C=CC1(C(=O)NC2CC3(CC3)C2)CCN(C(C2CCCCO2)=O)C1 N1(C(c2ccn(C)n2)=O)CC2(NC(c3cc(-c4ccncc4)ccn3)=O)CC1C2 N1(C(c2c(C)ncn2O)=O)C2CCC1CC(CCNC(=O)CSC(F)F)C2 c1(C(=O)NOCC(C2CCCN2)=O)ncnc2sc(Br)cc12 C1(NC(CNC(=O)OC)=O)CC2CC1CC2C(=O)NCC(F)C1CCC1 N1(C(CSC(C)=O)=O)CC2C(C1C(=O)Nc1cc(-c3ccc(Cl)s3)[nH]n1)C2(C)C CC1CN(C(C2(C#N)CC2)=O)CC1NC(=O)COc1ccccc1 c1(C(=O)NC(CCCCNC(C(CCC)(C)O)=O)C)cc(=NS(C)(=O)=O)cc[nH]1 c1(C(=O)NC2CCCC(NC(c3cc(C(C)C)on3)=O)C2)cnc(Cl)cc1N S(=O)(=O)(c1cc(C(=O)O)c(F)cc1OC)N1CCN(C(CC)C)CC1 Cc1cc(O)c(C(=O)NCC2(O)CCN(C(=O)COCC3CCCOC3)C2)nn1 c1(SCC(C(=O)OCC)NC(=O)CN)cccc(N2CCOC2=O)c1 c1(CC(N2CC3(CN(C(C(C)CC(N)=O)=O)C3)C2)=O)cccc2occc12 C(=O)(CCCC(C)(F)F)NC(C(C(C)C)NC(=O)COCc1ccncc1)C CCCC(O)C(=O)NCCCOCCNC(C1COC(=O)N1)=O Cc1cc(C(=O)NC2(CC(=O)NOCCCNC(N)=O)CCCCC2)c(C)cn1 CCCCCC(CC)C(=O)NCC1(C)CCCN(C(=O)CCOCC)C1 c1(NC)ccccc1C(=O)NC1(C)CC(NC(=O)CC(C)(C)SC)C1 N1(C(CC2C(OC)CC2)=O)CC(F)(CNC(c2cnc(-c3ccoc3)s2)=O)C1 N1(C(CCC2(C)CN(C(C(C(C)C)O)=O)C2)=O)CCCC(C)(C#N)C1 Cc1cnn(C)c1C(=O)NCC1(F)CC(NC(c2ccc(SC(C)C)cc2)=O)C1 C1(C(=O)Nc2ccc(SC)o2)CN(C(=O)CC(C)N(C)C)CCC1O c1(C(=O)NC23CC(CNC(Cc4cc(C)sc4C)=O)(C2)C3)c[nH]c2ncccc12 C=C(C)C(C)(C)C(=O)N1CC2CCC2(NC(c2ccc(=O)n(C(C)C)c2)=O)C1 c1(C(=O)NC2CC(O)(CNC(C(C)(C)C(N)=O)=O)C2)cccc2c1C1CCC2O1 N1(C(CC(C)SC)=O)CCCCC1CNC(c1ccc(CSC)o1)=O N1(C(C)C)CCC(C(=O)NC2CCCC(N(C)C(c3cn(C)nc3Cl)=O)C2)CC1 c1(CNC(CCC)=O)ccc(C(=O)NC2CCC2NC(=O)C(C)SC)cc1 C1(OC)CN(C(=O)CCC2CCCOC2)CC1NC(c1ccc(CSC)o1)=O N1(C(C(CC)CC(F)F)=O)Cc2ccnn2CC(NC(=O)C=C2CCOCC2)C1 Cc1nc(C(=O)NCC2CCC(NC(=O)CNC(=O)C3CC3)C2)ccc1[N+](=O)[O-] CCCCC(C)CCC(=O)NC(C)C(C)(C)C(=O)N1CCCC1C c1(C(N2CC(C)C(NC(=O)CC3CC=CCC3)C2)=O)cc2scnc2[nH]1 C1(CC)CCCC1(C)C(N1CC(C(=O)NCCNC(c2cc(F)n[nH]2)=O)C1)=O N1(C(c2c(C)coc2)=O)CCN(C(=O)CNC(c2c(C)n[nH]c2C)=O)CC12CC2 C1(NC(C2CCC(=C)CC2)=O)CCCC2CN(C(C3CC3C)=O)CC12 N1(C(C(C=C)(C)C)=O)CCCCC2(C1)CN(C(=O)C(C)(O)C(C)C)C2 CCCCC(CC)CC(=O)NC1CC(NC(=O)CN(C2CCC2)C)CC1O c1(C(=O)NCC(C)NC(C2CN(CC)C(=O)C2)=O)cnc2n(c1=O)CCS2 C(=O)(CCCCN(C(=O)C(CO)c1ccccc1)C)N(C)C.C1C(O)CC(=O)N1 c1(C(N(C2CCN(C(=O)C(C)CF)C2)CC)=O)ccc(N(C)C)nc1 C#CCC(C)(C(=O)N(CCC)OC)NC(C1(C2CCCO2)CC1)=O N1(C(C(C)P(C)(C)=O)=O)CC2CCC(C1)N2C(c1ccn(C2CC2)n1)=O CN=c1nc(N2CCCCC(C)C2)[nH]c(=NCC2CSCCS2)[nH]1 Cc1ccc(C(=O)NCC(N2CCC(C)C2C)=O)nn1 S(=O)(=O)(c1ccc(NCCN(C)CC2CC2)c(Cl)c1)NC1CC(C(C)C)OC1 c1(C(N(C(C)CNC(C2(C(=O)NC3CC3)CC2)=O)C)=O)c(Cl)csc1Cl C1(C(N(c2cccc(C(=O)OC(C)(C)C)c2)C)=O)CC(C(C)(C)C)=NO1 c1(N2CCN(C(=O)NC(C(F)(F)F)C3CC3)CC2)ncc2n1CCCC2 C(=O)(C(C(C)F)N(C)C(=O)OC(C)C)N(CCN(C(=O)CC1CC1)CC)CC C1(C(N2CC(OC(=O)NC)C2)=O)C(O)CCN1C(=O)CCc1conc1C CCCCCCCCNC(=O)C(N1CC(O)CC1CNC(C1CC1C(N)=O)=O)=O C(=O)(C1=NN(CC(C)C)C(=O)CC1)NC(CC)CN(C(=O)C1=CCSC1)C C1(CNC(CC=C)=O)CCCC2(CCN(C(c3cnn(CC)c3CC)=O)CC2)O1 C=CCCC(F)(F)C(=O)N(C)CC1CCCN1C(=O)C=CSC c1(C(=O)NC(CNC(C(CC#C)O)=O)CCOC)oc2c(C)cccc2c1C N1(C(C(CCOC)C)=O)CC(C(=O)NC(C)CC(C)(C)CO)CC1(C)C C1(C(=O)NCC2(C)CC(NC(C3C(C)(C)OC3(C)C)=O)C2)CC(C2CCCC2)C1 c1(C(C)NC(c2n(CCCCCC)nnn2)c2cnc(Cl)s2)c(F)cccc1F N1(C(=O)Nn2cccc2)CCCCC(Cn2cc(Cc3ccc(Cl)nc3)nn2)C1 CCCC(C)(C)C(=O)N1CCC(CC(C)NC(=O)C(C)(O)c2ccccn2)CC1 C1(COC(=O)OC(C)(C)C)CC12CCOCC2.C1(C(=O)OC)CC2C(C1)C(=O)N2 C1(NC(=O)CN(C2CCC2)C(c2ccc(O)cn2)=O)CCOC12CCOC2 c1(C(=O)NC2(CCNC(c3cncc(OC)c3)=O)CCC2)ccnn2ccnc12 C1(F)(C(=O)OCC)CN(C(=O)Cc2cc(C(F)(F)F)cc(F)c2)CC12CNC2 NS(=O)(=O)C1(c2cn(CC3CCCN3C(c3cc(O)ccn3)=O)nn2)CC1 c1(C(c2nnnn2CCSC)NC(C=C)(C)CC)ncn2ccccc12 C1(O)(CNC(C(C)OCC=C)=O)CC(C(N2CCC2(C)C(=O)OCC)=O)C1 c1(OC)cc(F)c(F)cc1C(N1CCC(NC(C2OCCC2C)=O)CC1)=O c1(NC(N2C(CNS(N)(=O)=O)CCCC2)=O)cnc2c(c1)CNC2=O c1(CC(=O)NCC2CCC(NC(CC(=O)NCC)=O)C2)ccc(C)nc1Cl c1(SC)c(C(=O)N(CCNC(c2ccccc2C(N)=O)=O)CCOC)cnn1C N1(C(C2(C)CCC2)=O)CC2CCC(NC(C3(C(F)(F)F)CCCC3)=O)CC2C1 C(C(=O)NCC1(F)CN(C(=O)CCC2CCCCN2C)C1)(C(C)(C)C)SC C(C(CCC)C(=O)N1CC(C)(C)C1C(C)C)NC(C(CCC)O)=O N1(CC(=O)NCC(CN(C(C(C)OCC#C)=O)C)(C)C)C(=O)CCC1=O Cc1nc(O)ccc1C(=O)NCCCCC1CCCN(C(c2cn[nH]c2)=O)C1 C(=O)(C1=CCCN(Cc2cc(C)nnc2O)C1)Oc1ccc(OC(C)(C)C)o1 C1(CC)CN(C(c2ccn(C(F)F)n2)=O)CCC1NC(C1(c2ncco2)CC1)=O Cc1ccccc1N1CCC(N(C)C(C2(N)CC3CC3C2)=O)C1=O c1(C(N2CCC(C)(CNC(C3ON=C(CC)C3)=O)CC2)=O)ccc2sccc2c1 C1(OC)CCC(NC(=O)C(F)(F)c2cccnc2)C1.C1CC(=O)N2CC(C2)S1 CC1(C)CN(C(c2ccccc2OC(F)F)=O)CCC1NC(C1CCC(F)C1)=O CC1CCCC=C1C(=O)N1CC(O)CC1CNC(c1ccc(Br)cn1)=O C=CC1CN(C(=O)CN(C)C)CC1NC(=O)CSc1ccc(Br)cc1 CCC(C)CC(=O)NC1CCC(NC(c2ccccc2C(=O)NCCO)=O)CC1 O(NC(=O)C(CNC(=O)CC1CCC(=O)N1)CC(C)C)C(CC)CC N1(CC(N2C(CNC(c3cccn3C)=O)CC(OC)C2)=O)C(=O)CC(C)(C)C1=O c1(C(c2n(CCCSC)nnn2)NCC2(C(F)(F)F)CCC2)noc2c1CCC2 N1(CCC(=O)NCC(=O)N(CC#N)CC#N)CCOCC1 Cc1noc(Cl)c1CC(=O)NCCC1CCCN1C(=O)C(C)CO C(C)(C(=O)NC(C(=O)NCC1(C(F)(F)F)CC1)C1CCCC1)OC(C)=O C1(CCNC(C(n2c(C)ccn2)C)=O)CN(C(c2csc(F)c2)=O)CC1C c1(CCOC)sc(C(=O)NC2CC(F)(CNC(=O)CCc3cnc[nH]3)C2)cc1C N1(C(c2ccc(C)s2)=O)CCC(C)(C)CC1C(=O)NCC1(C)CCCO1 C=CCC(O)(CC=C)C(C)NC(=O)Nc1ccccc1CNC(C)=O CCCCS(=O)(=O)CC(=O)NC(CNC(c1cnc(C(N)=O)cn1)=O)CCOC c1(OC)cc(Br)c(F)cc1S(=O)(=O)Nc1ccc(F)c(CCC(=O)O)c1 C(CCCCCN=[N+]=[N-])NC(C1CC(C(C)O)C1)=O c1(C(=O)NC2C(C)CN(C(C3CCC3)=O)C2)ccc(-n2cncn2)c(F)c1 C(=O)(C(CCC)C(C)C)N(CC(=O)NC(CC#C)CCOC)CCOC Cc1cc(C#N)cnc1C(N1CCC(C)(C)CC1C(N1CC2CC1CS2)=O)=O C1(C(=O)NC2C3CN(C(=O)CCSC(F)(F)F)CC23)CCC2(CCC2)C1 C(=O)(C(=O)C(C)(C)C)N(CCC(=O)N(C)Cc1c[nH]nc1C)CC#C CC(C)(C)C(=O)CCC(=O)NC(C)(C)CCCNC(C1CCN1C(C)(C)C)=O c1(C(=O)NC23C(CN(C(COc4cccc(C)c4)=O)C2)C3)cscc1S(C)(=O)=O C12(NC(=O)COc3ccc(F)cn3)CCCCC1N(C(c1ccc(Cl)s1)=O)CC2 N1(C(C=CC)=O)CCN(C(c2cc(C)co2)=O)CC1C1CCCC1 c1(OC)ccccc1-n1nc(Cc2cscn2)nc1-c1ccc(C)n1C c1(CNC(C23C(CN(C(=O)CSC4CC4)C2)C3)=O)nc2ccccc2s1 C(=O)(CCS(=O)(=O)CC(C)C)NCC1(CNC(c2cccc(C)n2)=O)CC1 C1(O)(CNC(C(CC)C)=O)CCCN(C(=O)CC2(N3CCCC3)CC2)CC1 CCC(C)(CNC(=O)C(=CC1CCCC1)C)NC(c1cn(C)nn1)=O c1(OC)cc2c(cc1Br)C(NCCc1ccc(C)c(Br)c1)CC2 N1(C(C=C(C)Cl)=O)C2CCC1CN(C(c1cc(O)c(F)cc1N)=O)C2 C(C(=O)NCC1CC1CNC(=O)Cc1ccnnc1O)(C(C)(C)C)OC Cc1cc(Cl)c(C(=O)NCC2CCC(C)CN2C(c2cnsc2)=O)cc1F CCC(CC(=O)N1CCC(C(N2CC3(CSC3)C2)=O)C12CCC2)C(C)C c1(OC)c(C(N2CCC23CN(C(c2occc2C)=O)C3)=O)cnc2ccccc12 c1(SCC(=O)NC(C2N(C(C(CC)NC(C)=O)=O)CCC2)C)cccc(OC)c1 N1(C(c2c(CC)[nH]c(=N)s2)=O)CC2CN(C(C3CC(C)(C(=O)OC)C3)=O)CC2C1 c1(CC(N2C3CN(C(CCCCOC)=O)CC2C3)=O)c(C)nc2ncnn2c1C N1(C(c2c(CC)ncnc2)=O)CCC(O)C(NC(=O)C(C(C)C)C2CCC2)C1 c1(CCC(N2CCC(CNC(C(C)C(F)F)=O)CC2C)=O)cnc2n1CCOC2 c1(C(=O)NCC(C)C(N2CCCC(N(C)C)CC2)=O)ccc(F)c(F)c1 C(c1ccsc1Br)=CC(=O)N(CC(C)NC(CCCOC(C)C)=O)C O=C(CC1=Cc2ccccc2C1)NC1CC1c1ccccc1 c1(C(=O)NCC(C2CC2)NC(=O)CCCN2CCCCC2)cnc2c(c1)CCC2 CCC(C)CCCC(=O)NC(C(=O)NCc1cc(C)ncn1)C1CCC1 c1(OC)ccc2c(C)cc(-c3ccc(C(=O)NC4CCSC4)cc3)nc2c1 c1(C(N(c2ncc(C(=O)OCC)cn2)C2CCCN2)=O)cnc2cc(C)ccn12 c1(-c2cn(CC3CN(C(c4cc(C(F)(F)F)co4)=O)C3)nn2)cnc(Cl)c(Cl)c1 N=c1ncc(C(=O)NCC2(O)CN(C(C3CCCC(O)C3)=O)C2)c[nH]1 c1(C(=O)NCC23N(C(c4csc(C)c4N)=O)CCC2CC3)cc2cccnn2c1 C1(C(CO)NC(CC2CCN(C)C2)=O)CCN(C(c2ccn(C(F)F)n2)=O)CC1 C(=O)(CCC(C)S(C)(=O)=O)N1CC(n2cc(CNC(C(C=C)O)=O)nn2)C1 CC(C)C(CC(=O)NCC(C)(C)C(C)O)NC(=O)CC1CCC(=O)N1C C(c1ccc(Br)cc1)=CC(=O)NC1CCN(C(C2CCOC2)=O)CC1CO C#Cc1cn(C)nc1C(=O)NC1(CCNC(=O)C(O)C2CCCC2)CCC1 Cc1sccc1C(=O)NCC1(C(C)NC(C23CC(F)C2C3)=O)CC1 C1(NC(C2(OC)CCC2)=O)CCN(c2ccnc(Cc3ccccc3)n2)CC1F C(=O)(CC(C)(C)C#N)NCC(CN(C(C1CCC(C2CC2)C1)=O)CC)(C)C N1(C(C(C)(C2CC2)OC)=O)CCCC2(CCN(C(=O)CSc3n[nH]c(O)n3)C2)C1 C1(CC(=O)NCC(CN(C(CC(C)F)=O)C)(C)C)CC(C)(C)CO1 CN1CCC(n2nccc2-c2ccc(N)cn2)CC1.N12CCC(C1)CC2=O c1(OC)nc(Cl)ccc1C(=O)NC1C2CC1N(C(=O)CSCCC(F)(F)F)C2 CC(C)(C)CCC(=O)NC1CCCC(NC(c2ccsc2C#N)=O)C1 c1(N2CCC(CNC(c3ccc4nn[nH]c4c3)=O)C2)ncnc2cnccc12 N1(C(CNS(CC)(=O)=O)=O)CCCC(C)(C)C1CNC(C1CCCCC1(C)C)=O C1(C(CNC(C(CC)C)=O)O)CCN(C(c2cncn2C2CC2)=O)CC1 C1(CCC)CN(C(=O)C(O)CC(F)F)CCN1C(=O)C(F)CC N1(C(c2cnn(C)n2)=O)CC(C(=O)NC2(CO)CC3CCCC23)C(F)(F)C1 C(=O)(C(CC)C(C)OC(c1ccccc1-c1ccccc1)=O)OCC c1(C(N2CC(C)C(CNC(c3[nH][nH]c(=N)c3Br)=O)C2)=O)cnc2n1CCOC2 C(=O)(C1=CCCN(C(c2cn3c(n2)CCC3)=O)C1)NC1CC(C)(C)OCC1 C12(CC(N3CCC(COC)(NC(=O)C=C(C)Cl)CC3)=O)CCC(CC1)C2(C)C C12(C(=O)Nc3c(N4CC(C)OCC4)ccc(F)c3)CC(C)(C1)OC2(C)C c1(C(N(CCn2cc(CSC)nn2)CC)=O)cc2ccc(OC(F)(F)F)cc2[nH]1 C(CSC)(C(=O)N1CC(F)(C(=O)NC(CC2CC2)CO)C1)OC c1(CC(=O)NCC2CC3CCC2C3)cc(F)cc(F)c1.C12(F)CCCN(C1)C2=O N1(C(c2ccn(CC)c2C)=O)CCN2C(=O)C(NC(c3cc(C)c[nH]3)=O)CC2C1 C(N(C)N1CCCN(c2ccncc2)CC1)c1c(CC)onc1C c1(C(N2C(CN(C(C3C(CC)C3)=O)C)CCC2)=O)ccc(F)c(CSC)c1 c1(C(N(CCN(C(=O)CSCc2cccs2)CC)CC)=O)n[nH]c2c1CSCC2 c1(C(N2C(CN(C(C(COCC)(C)C)=O)C)COCC2)=O)c(F)cc(C)cc1F c1(OC)ncc(CN2CC(OC)CC2C(N2CC3CC2CO3)=O)cn1 C(=O)(C(C)(F)C(C)(C)F)N1CCCC(NC(Cc2ccc(OC)nc2)=O)(CO)C1 c1(C(C)NCCc2nc(C(C)C)sc2)cc2n(n1)CCCC2 n1(CC)ccnc1C(C)NC(C(C1CCC(C)C1)N(C)CCC(F)F)=O c1(C(=O)NCCCCNC(=O)C(O)CF)ccc2c(c1)OCC2 C#CCCCCC(=O)NCCCNC(c1cc(C2CCC2)no1)=O c1(C(N2CC(CCC#C)C2)=O)ccnc(CNC(c2ccnc(CC)c2)=O)c1 C(=O)(C#CC1CCC2(CC1)OCCO2)N1CCCC(O)(CNC(C(C)C)=O)C1 C1(C(=O)NCC2CCCO2)CSCCN1C(c1ccc(C2CC2)o1)=O CC(C)C(C(=O)NCCCCCNC(c1ccnnc1S)=O)NC(N)=O C(C(C)(C)CN(C)CC)NC(CCN(C(=O)CC1CC=CCC1)CC)=O N1(C(C2(COC)CCC2)=O)CCC(CN(C(=O)C(C)CF)C)CC1 C1(C(=O)OC)CC(F)(F)CN1C(c1ncc(Br)cc1F)C(=O)NC1CCC1 CCCCCCCC(=O)N1CCCC1(C)CNC(=O)Cn1ncnn1 n1(CCCC)ncc(C(N2CCCC2CCCNC(C2(C)C=CCC2)=O)=O)c1C CN1CCC(F)(CNC(C2CN(C(c3c[nH]cc3C3CC3)=O)CCO2)=O)C1 c1(C(=O)OC)cc(C(N2CC(NC(c3cn[nH]c3)=O)C(O)C2)=O)ccn1 C1(O)(CC)CN(C(=O)C(CC2CCCC2)NC(=O)Cc2ccc[nH]2)C1 N1(c2nc(Cl)nc(CC)c2Cl)CCC(C2CCCN(C(=O)CC3(O)CCC3)C2)C1 C1(C(N(C)CC2CCSC2)=O)C2CCN(C(C3CCCC(C)(C)C3)=O)CC12 C1(C(=O)NC2CC2O)(COC)C=CCN1C(=O)CNc1ncccn1 C1(C(N(C2CCN(C(=O)C=CBr)C2)C)=O)CC(O)CN1CC(F)(F)F c1(C=O)cnn2c1CN(C)CC2.c1(C(=O)NCCN(CC)CC)cccc(CF)c1 C1(C(=O)OC)CCOC1C(=O)NC1CCN(CCOC)C1 n1(CC)ccc(C(=O)NCC2COCC2NC(=O)C(c2ccc(F)cc2)F)c1C c1(C(N2CC(CNC(c3cnc4ccoc4c3)=O)C2)=O)c[nH]c2cccc(Cl)c12 N1(C(C(C)SCCCC)=O)CC(CC(=O)NCc2snnc2C)C(C)C1 c1(C(N(CCCN(C)C(C)C)C)=O)coc(C(F)F)n1.C1(=O)CCO1.CC(F)F N1(C(c2ccsc2C(F)F)=O)CCCC1C1CCCN1C(=O)Cc1cnns1 C(=O)(CC(C)(C)CC(F)F)NC1C=CCN(C(c2cc(C)nn2C2CCC2)=O)C1 C(=O)(C1=CCCCCC1)NC1(C)CCN(C(C2CCCC2P(C)(C)=O)=O)CC1 c1(C(=O)Nc2nnc(C)o2)ccc(-c2csc(-c3nc[nH]n3)c2)cc1 CC1(CNC(=O)C(F)(F)c2ncccn2)CC(NC(C2CCCCS2)=O)C1 N1(C(CCCSC)=O)CCN(C(=O)C(C2CC2)C2CC2)CC2CCCCC12 C1(NC(c2cc(CC)no2)=O)CN(C(C2CC3(CC3)CO2)=O)CC1C n1(C(C)(C)C)cc(CNC(c2cnn3c2OCC3)=O)c(O)nc1=O C(C)(C)(CCC(=O)NCCC(O)CNC(C1C2CCCCCC12)=O)N(C)C C1(C)(CNNC(CC2(N(C(CC(C)C)=O)C)CC2)=O)C=CCCC1 N1(C(C=C(CCC)C)=O)CC(C(=O)NCCC(=O)N(C)C2CC2)C(F)(F)C1 C12CCC(CC1)C(=O)NC2.C(CC(=O)N(C1CCC1)C)OCCSC CC1CC(OC(=O)C(c2ccccc2)C2CCCCC2)CC(C)C1 c1(OC)ccn2c(C(=O)NCCC3(NC(c4cnco4)=O)CC3)cnc2c1 c1(CC)nc2c(C(N3CCN(C(c4cn(CC)cn4)=O)CC(O)C3)=O)ccnc2[nH]1 C1(NC(C(c2ccc(OC)cc2)CC)=O)CCN(C(=O)CCC#N)CC1O c1(C(=O)NC2CCC3C(C(=O)O)C32)ccc2nncn2c1 N1(C(c2cc(C)no2)=O)CCCC(CC(=O)NC2CC2c2ccccc2)CC1 CC(C)(C)C(C)(O)C(=O)NC1(CNC(C2CC(n3cnnc3)C2)=O)CC1 CC(C)CC(C(=O)N(CCCNC(=O)C(C)(C)C(C)C)CCO)n1ccnc1 c1(C(=O)NC(C)CN(C)CC2(O)CCSC2)nnn(C)n1 CCC(C)(CCNC(=O)CC1CCCS1)NC(c1ccsn1)=O c1(C(=O)NC2CC(NC(C3CCOC3c3cn[nH]c3)=O)C2)cccc(C(F)F)c1 CCC(C(=O)N1CC(CCNC(C2CCCSC2)=O)C1)n1ccc(C2CC2)n1 c1(-c2n(-c3c(C)cccc3)nc(CCCO)n2)ccc2ccccc2c1 c1(CC(=O)NCC(C)(C)CNC(=O)CC2CCOC2=O)cccc(Cl)c1 c1(OCc2nnc(COC)s2)cc(N2CCCCC2)cc(Cl)c1 c1(-n2cc(C3(NC(C4OCCCC4(C)C)C)CCC3)nn2)ccc(Br)c(Cl)c1 N1(CC)CCCC1CC(=O)NCCCCN(C)C(c1sncc1Br)=O C1(C(CC)C)CCC(C(N)C2CC2)CC1.C(=O)(NC)OC N1(C(Cc2[nH]c(=N)sc2)=O)CCOC(CCNC(C2CCCC2(F)F)=O)C1 C1(CNC(C(CNC(CCC)=O)OC)=O)CCCCC1CC C(CCCc1ccccc1)(C(=O)OC)NC1(CCOC)CC1 C1(CNC(c2cnc(SC)s2)=O)(CNC(=O)Cc2cccnc2)CC12CCC2 C(=O)(C1=CCCCO1)NC(C(=O)NC(c1ccccc1)CC)CCC1CCC1 C1(NC(=O)OC)CCCN(C(C(=O)Nc2ccc(OC)cc2)C2CC=CC2)C1 c1(C(N(CC(C)NC(=O)Cn2nccc2C)CC)=O)ccc(C)c2ccccc12 C1(CCCNC(c2nc(CCC)sc2)=O)CCN(C(=O)Cc2cn[nH]c2)CC1 C(=O)(C1CCCc2nnn(C)c21)N1CCCC(N(C(=O)CCCC#N)CC)CC1 N1(CC(=O)NCCC2(O)CCCN(C(CCC#CC)=O)C2)CCc2sccc2C1 Cc1nn(C(C)C)c(NCC2(F)CC(NC(C3CC(=O)N3)=O)C2)c1[N+](=O)[O-] c1(C(N(C(CCNC(c2cc(C)on2)=O)C)C)=O)coc2c1COC2 c1(C(N2C(C(=O)NCC3N(CC)CC3)C=CC2)=O)ncnc(O)c1F n1(CCC(C)C)c(C2(CN(C34CCCCC3C4)C=O)CC2)nc2ccccc12 N1(C(c2cc(OCC)ncc2)=O)CCC(O)(CNC(c2conc2CC)=O)CC1 N1(S(=O)(=O)CC2(CF)CCOCC2)CCC2(CC=CCO2)CC1 c1(NC(c2c(F)cc(Br)cc2F)c2n(CCC)nnn2)ccc2nn[nH]c2c1 c1(C(C2CN(C(CC)=O)C2)C)cn(Cc2conc2C(C)(C)C)nn1 CCC(C(=O)N1CCN(C(=O)C=Cc2cn(C)nn2)C(CO)C1)C(C)(F)F Cc1cc2[nH]c(C(=O)N(C(C)CCNC(c3cc(S(N)(=O)=O)c[nH]3)=O)C)cc2o1 Cc1cccc(C(N2C(C(=O)O)CCC2(C)C)=O)c1[N+](=O)[O-] C(=O)(C(C)CCC(C)(C)C)NCC1(OC)CN(C(=O)CNC(=O)C(F)(F)F)C1 c1(N(C2CC(OCCCC)C2(C)C)C)ccc(I)c(F)n1 c1(CC(=O)NC(CCCNC(c2n(C(C)C)ncn2)=O)C)ccccc1O N1(C(C2CCN(C(C3CCC(C)O3)=O)CC2)=O)CCN(C)C(C2CC2)C1 c1(C(=O)NCC(CNC(c2[nH]cc(C(=O)OC)c2)=O)OC)ncn2c1CCCC2 c1(N2C(CCCNC(c3c(CC)ncs3)=O)CCC2)ncnc2c(Br)cccc12 N1(C(CC(C(CC)C)NC(=O)C(C)N=[N+]=[N-])=O)CCN2C(=O)CCC2C1 N1(C(CNC(CC)=O)=O)CCC(C)(CNC(=O)C(N2CCSCC2)C)C1 C(C(C(=O)NC1CC(CC)C1)n1cc(CN2CCCC2)nn1)OCC C1(C(N2CC(C)N(C(c3ccnc(Cl)c3N)=O)CC2)=O)CCC2(C1)CC2(F)F c1(CC)cncc(C(N2CC(NC(=O)CCN3CCN(C(=O)OC)CC3)C2)=O)c1 CS(=O)(=O)CCC(=O)NC12CCC(C(=O)NCC3CC(O)CCO3)(CC1)C2 C1(C(N(CCCC(=O)NCC(=C)Br)C)=O)C(C)(C)C1(F)F c1(C(N2CCCC(O)(CNC(Cn3c(C)cnc3)=O)C2)=O)ncnc2sccc12 c1(CC)ccc(CC(=O)N(C2CCCN(C(C3CCCO3)=O)C2)CCO)cc1F C1(C(=O)NC(CC)CO)CC(F)(F)CN1C(c1ccnc(C)n1)=O C1(CC(=O)NC(C(=O)N(CCC=C)CC)C2CCC2)CC(C)(C)CO1 Cc1ccc(C=CC(=O)NC2CCC(CNC(=O)CCc3nccs3)CC2)nc1 Cn1cc(C(=O)N(CCC(C(C)(C)C)NC(=O)C=CC=C(Cl)Cl)C)n(C)c1=O C(=O)(C(CO)C(F)(F)F)NC(c1c(C(N(C(C)C)CCN(C)C)=O)con1)C N1(c2c(C)coc2C#N)CCCN(c2nc(-n3ccc(O)nc3=O)ns2)C(C)C1 c1(C(N(C)CC2CCCCN2C(c2cnc[nH]2)=O)=O)cc(F)c(F)cc1O C1(C(N2CCN(CC(N)=O)CC2)=O)CCCCCN1C(=O)C(F)OC(F)(F)F N1(C(c2c(OC)cccc2O)=O)CC2(CCN(Cc3cccc(O)c3Br)C2)C1 C1(C(=O)NCc2cc(CC)no2)CN(C(c2ccoc2C2CC2)=O)CC(C)(C)C1 O(NC(=O)CCCCC(C)C)C(C(=O)OCC=C(C)C)C c1(CN2CCC(C)(NC(c3c(C)cccc3)=O)C2)cccc2[nH]ncc12 C1(C(=O)NCC(CNC(C=Cc2cn(C)nn2)=O)(C)C)CC2(C1)CC(O)C2 c1(C(=O)NCC2N(C(c3ccc(C(C)=O)cc3F)=O)CC2)coc(S(N)(=O)=O)c1 c1(C(=O)NCCOC2CCN(C(c3c(C)n(C)nn3)=O)C2)cc(Cl)c(Cl)n1C Cc1cc(CC(N2CC3CC(NC(C4C(F)(F)C45CCC5)=O)C2C3)=O)cc(F)c1 C(=O)(C1COc2ccccc21)NC1CCCC(NC(c2cc(C)nc(O)c2)=O)C1 C(=O)(NNC(=O)c1ccn(CCC(C)C)n1)c1n(C(C)C)cnc1 N1(C(c2noc(C)c2C)=O)CC2CCN(C(c3cncc(F)c3)=O)CC2C1 C(=O)(CCCC(N)=O)NCC1N(C(C2CCC(C)(CC)O2)=O)CC(F)C1 N1(C(C2OCC(C)(C)C2)=O)CC2(CCCC2NC(=O)COCc2nc[nH]n2)C1 C(=O)(CC(F)(F)C(C)C)N1CCC(CNC(C=Cc2c(C)noc2C)=O)C1(C)C CCCC(C(O)C(=O)NCCCC(C)CO)NC(c1cccnc1)=O c1(C(=O)NCCCC(C)NC(c2cccn2C2CC2)=O)cc(C(F)F)ncn1 CC1(C)OCCC1CC(N1CC2C(CC(=O)NCC(C)(C)OCCO)C2C1)=O C(=O)(C1=CCCCC1C)NCC(CCC)C(=O)NCCC#CCO c1(N(C)C)ncc(C(N2CC(CNC(=O)C(=O)NCC(F)(F)F)C2)=O)cn1 C1(C(=O)NCCNC(c2cc(C)on2)=O)CC2CCC(C1)N2c1cnccn1 c1(CC)ocnc1C(=O)NCCCC(C)NC(=O)Cc1cnn(CC)c1 C=CCC(CC(C)C)C(=O)N(CCCCCC(=O)N(CCO)CC)C CCCCC(CC(=O)NCCCC(C)(C)OC)NC(=O)C(C)(O)C1CC1 C1(C)(C(C)C)CCN(C(=O)NC2CCCC2c2ccc(Cl)cc2)CC1 C12(CNC(C3(NC(c4occ(C)c4)=O)CC3C)=O)CCC(CC1O)C2 Cc1cc(CNC2CCC(C(=O)NCCc3ccc(Br)cc3)C2)c(C)cc1O N1(C(C23C(CN(C(c4ccc(CCO)cc4)=O)C2)C3)=O)CCN2CCCC2C1 Cc1ccc(NC(c2ccc(NC(C34CCCC3C4)=O)nc2)=O)cc1F C#CCCCCCC(=O)N1CC(NC(C2(C)CCN(C)C2)=O)CC12CCC2 c1(CC)cc(F)ccc1C(=O)NCC1CCN1C(=O)CNC(C1CCCC1)=O N1(C(C2N(N=O)CCC2)=O)CC2CC(C1)CN(C(=O)CCc1ccco1)C2 C(c1cccc(Cl)c1)=C(C(=O)NC1CCCN(C(c2n(C=C)nnc2)=O)C1)C C1(C(=O)NCC2N(C(CCC(C)(F)F)=O)CCC2)CC2COCC(C1)C2 c1(OCC)ccc(Br)c(C(F)(F)F)c1.c12cc(cc(F)c1)CNc1ccc-2nc1 Cc1ccc(OC(F)(F)F)c(C(=O)NC2COCC2NC(c2ccc(Br)o2)=O)c1 c1(C(=O)NC(CNC(C(CC)(C)C)=O)C(C)C(C)C)cncc2c1CCNC2=O C(=O)(CCCC(F)(F)CO)N1C(CN(C(CCC(CC)OC)=O)C)CCCC1 Cc1cc(F)ncc1CN1CC2C(C(=O)Nc3ccc(Br)c(F)c3)C2C1 c1(C(N2C(C(C)NC(C3(COC)CC(=C)C3)=O)CCC2)=O)ncc(C)cc1C c1(CC(=O)NC(C(C)NC(CN(CCC)C)=O)C(C)C)ccc(F)c(OC)c1 CC1OC2CCC1(NC(=O)C=CCC(C)(C)NC(=O)CCCCC1CC1)C2 C#Cc1ccc(C(N2CCC(C(=O)NCC3(OC)CCSC3)C2)=O)c(C)c1 C1(C(N(CC(C)(C)NC(CC(=O)NCC)=O)C)=O)CC2CCC1NC2=O N1(C(C2(CCOC)CC2)=O)C2CCC1C(CNC(c1scnc1Cl)=O)C2 CS(=O)(=O)c1cccnc1C(=O)NCC#CCNC(=O)CN1CCSCC1 c1(C(N2CCC(CNC(C3C4CC5C(C4=O)C35)=O)CC2)=O)cc(F)cc(F)c1 Cc1cccc2c(=O)c(C(N3CCCC(CO)(NC(=O)CC(C)F)C3)=O)c[nH]c12 C1(CC)CCC(CNC(C2(NC(=O)C=Cc3nccs3)CC(F)C2)=O)O1 n1(CC(=O)N(CCC(C)NC(C2CCC(NC(N)=O)CC2)=O)C)cnc(C#N)n1 N1(CC(=O)O)CC2(CCN(CC3CCCN3C3CCCCC3)CC2)OC1=O Cc1cc(F)ccc1C(F)(F)C(=O)NC(C)CNC(=O)CC1C(=O)N(C)N=C1C CCC(C)C(CNC(=O)CC(O)CNC(=O)CC(C)c1ccco1)CO C=CC(C)CC(=O)NCC(c1cccc(OC)c1)NC(=O)C1=CSCS1 C1(C(=O)NC(C)CCNC(=O)CCCCCNC(N)=O)CS(=O)(=O)CC(=O)N1 Cn1c(C(N2CCC(CCNC(=O)CC(C)(C)C3CC3)CC2)=O)nnc1S CC(C)CC(=O)C(=O)NCC(C(=O)NCC1CCC(O)CC1)N(C)C Cn1c(C(N2CC(F)(F)CC2CCNC(=O)CC2CC23CC3)=O)cccc1=O c1(C(C(=O)NCCOC)N(CCC)C)n[nH]c2cc(OC)c(OC)cc12 N1(C(CC(C)C2CC2)=O)CCCC(O)(CNC(c2cnn3c2N(C)CC3)=O)CC1 C1(C(NOCc2cccc(C)n2)=O)CCCCCN1C(C1CN(C)C1)=O c1(C(N(CCNC(c2cncc(C)c2)=O)C)=O)c(C)nc2sc(C)nn12 C1(NC(NC(c2ccccc2)C)=S)CCC(c2ccccc2)C1 c1(NC(CC2(NCc3ccc(SC)s3)CCC2)=O)ccc(C)nc1N1CCCC1 N1(C(c2c(CNC(c3c(C)nc(CC)o3)=O)nnn2C)=O)CCC(C)CC1CC C1(C(=O)NC2(C(N(C)CC3CC3C3CCCO3)=O)CCCC2)CC(=O)OC1(C)C Cc1nn(C)cc1CNC(=O)C(c1ccco1)NC(=O)CC1CCOC1=O CC(F)(F)C(F)C(=O)NCC1CCN(C(=O)C(C)(O)C2CCC2)CC1 N1(C(c2c(COC)cco2)=O)CCN(C(C2CCC(OC)CC2)=O)CC(O)C1 C(c1ccc(C(N)=O)cc1)=CC(=O)NC(C1CN(C(C2(C)ON=C(C)C2)=O)C1)C c1(C(=O)NCC2C(NC(C(C)O)=O)CC2)cc2c(s1)CC(C)(C)C2 N1(C(C(=O)NC)=O)CCC(n2cc(CNC(C3CC(C)(C(=O)O)C3)=O)nn2)C1 CC(C)C1=NOC(C)(C(=O)N(C)Cc2ccccc2CNC(=O)CCC2CC2)C1 N1(C(c2c(SC)ccc(N)c2)=O)CC2(CCN(C(c3cc(Br)n[nH]3)=O)C2)C1 C1(CN(C(C(N2CCOCC2)C)=O)C)COCCN1C(C1CCCN1C1CC1)=O C1(C#CC(=O)N2CCC(CCN(C(=O)CC(C)OC)C)CC2)(CC)CC1 c1(C(=O)NCC(CO)N(C(=O)CCCCNC(N)=O)C)ccn2cncc2c1 CC1CN(C(C2CC2c2cccc(-c3ccc(Cl)nc3N(C)C)c2)=O)CCC1=O C(=O)(C1=NOC(C2(O)COC2)C1)N1CCC(CCC)C1 N1(C(c2c(C)cco2)=O)CCCCC1CCN(C)C(C1CC(F)(CO)C1)=O N1(C(c2c(C)[nH]cc2)=O)C2CCC1CN(C(c1cnc(C(C)C)n1C)=O)C2 c1(-c2c(C)nc(CC)s2)ccn2ncc(C(=O)Nc3cnc[nH]3)c2c1 N1(C(C2CNC(=O)N2)=O)CC2OCCN(C(=O)Cn3cnc([N+](=O)[O-])n3)C2C1 CC(C)C(O)CC(=O)N1CCC(NC(=O)CCCc2cccnc2)C1C c1(C(c2nnnn2C(C)C)NC(CCSCC)C)c(F)cc(C)cc1F CC1(C(=O)NCC2(CNC(=O)C(O)(C3CC3)C3CC3)CC2)CC=CCC1 c1(N2C(C)C(NC(=O)CCn3cnnn3)CC2)cc2c(cn1)C(=O)CCC2 Cc1c(C(=O)NCC(CCl)Oc2cccc(F)c2)ccn1C c1(OC)cc(OC)c2cc(C(=O)NC3CC(NC(C4CCC(C)C4)=O)C3)[nH]c2n1 C(c1cccc(F)c1)=C(C(=O)NCCN(C(c1c(CC)nc[nH]1)=O)C1CC1)F Cc1cnc(Cl)[nH]c1=NC1CCCOC1C1CCN(C(C2(F)CCOC2)=O)CC1 C1(CCCNC(Cc2n(C)ccc2)=O)CCN(C(=O)CCc2cc[nH]n2)CC1 Cc1cncc(C(=O)NCCCC(C)NC(=O)COc2c(C)cccc2Cl)c1Cl C(=O)(C1CCCc2c1ncn2C)N1CC(O)(CNC(c2n(CC)cc(Cl)c2)=O)C1 S(=O)(=O)(CC(=O)NCC1CCN(C(c2ccc(NC(C)=O)s2)=O)C1)NC c1(C(=O)NC(CNC(C2CCN(CC)C2)=O)C(C)C)cncn(C)c1=O N1(C(c2ccc(COC)s2)=O)CC2(CCCCN2C(=O)CN2CCCC2C)C1 Cc1nc(CC(=O)NC(C)(CNC(=O)CC(O)C2CCCC2)C2CC2)co1 C1(C(N2CC(F)(CO)C2)=O)CC12CCN(C(C1CCCOCC1)=O)C2 C1(NC(C2N(C)C(=O)CC2)=O)CN(C(=O)CC2C=CS(=O)(=O)C2)CCC1(C)C N1(C(C(CCC)F)=O)CCN(C(c2nnsc2C)=O)CC(C)C1 C1(C(N2C(CC(=O)NCCN(C)CC)CCCC2)=O)CC2(CCCO2)C1 C1(NC(C(C)N(CCC)C(c2coc(SC)c2)=O)=O)CC(C)N(C)CC1C C1(NC(C)=O)CCN(C(=O)COC2CC(NC(c3ccsc3)=O)C2)C1C N1(C(CC2CC(SC)C2)=O)CC(C2(NC(c3n[nH]c(C)n3)=O)CC2)C1 C(=O)(C(C)(F)C(F)(F)F)N(CC(c1ccccc1Br)O)C C1(NC(C2C3CN(C(=O)Cc4cc[nH]c4)CC23)=O)CCCC(C2CC2)C1 n1(C(C)C(=O)NC(C)(CNC(c2cnn(CCO)c2)=O)C2CC2)cnc(C#N)n1 C1(CNC(CCN(CCC)C)=O)CCCCN1C(=O)C(=Cc1c[nH]cn1)F c1(OC)ccc(O)c(NC(C2(F)CCN(Cc3c(OC)cccc3C)C2)=O)c1 n1(C(CC)CC)nc(C(=O)NCC(C)(C)CCNC(c2cnc(O)s2)=O)cc1C c1(C(N2CC(CC)N(C(=O)C(O)C(C)(C)C)CC2)=O)cc(N(C)C)cc(C#N)c1 N1(C(CC(=O)OC)=O)CC2CCC(C1)N2C(=O)CC1CC1C(F)(F)F C(=O)(C(C)C(C)(F)F)NCC(CCC)NC(=O)CC12CCC(CC1)C2 C(=O)(C(O)CC(N)=O)N(C(C(N1CC(C)(COC)C1)=O)(C)C1CC1)C c1(CC(=O)N(CCNC(COCCC=C)=O)C(C)C)cn[nH]c1 C1(OC)CN(C(c2sccc2-c2cn[nH]c2)=O)CC1NC(=O)CCF CC1=C(C(=O)NC(C)C(C)NC(c2c(OC(F)F)cccc2Cl)=O)CCCC1 N1(Cc2n(CCC)nnn2)CC2(CC(NC(c3c(C)nn(C)c3Cl)=O)CO2)C1 c1(C(N(CC(CC)NC(=O)CSC2CCS(=O)(=O)C2)C)=O)cncc2c1CCC2 c1(N(C(NNC(c2ccc(C)c(F)c2)=O)=O)Cc2ccsc2)cc(F)c(Br)cc1F c1(C2C(NCc3n[nH]c(-c4cccc(C)c4)n3)C2)ccc2c(c1)OCO2 CS(=O)(=O)C1CN(C(=O)CCCCc2cnn[nH]2)CC1NC(c1cc(F)n[nH]1)=O N1(C(C2CN(CC)C(=O)C2)=O)CCC(NC(=O)CSc2nncs2)C(C(N)=O)C1 c1(CCCN(CC(C)N(C(=O)CO)C)C)ccc(Br)cc1.C1(CS)CCCCO1 N1(C(C(C)NC(C)=O)=O)CC2=C(C1)CN(C(c1cc(C(C)C)[nH]c1C(C)C)=O)C2 Cc1ccc([N+](=O)[O-])cc1SCCCOc1cc(C)c(Cl)c(C)c1.C1CCN1C c1(OCCCC(=O)Nc2c(CNC(=O)COCCF)ocn2)ccc(F)cc1Cl C(=O)(C1CCCc2cccnc21)N(C1CCN(c2cc(C(N)=O)nc(Cl)n2)C1)C Cc1nc(Cl)ccc1CC(=O)NCC1CN(C(=O)CN2C(=O)CCC2=O)CC1O N#CC1=C(C(=O)N2CC3CCC3(CCNC(C3(CF)CCC3)=O)C2)CCC1 Cc1cc(C(=O)NC2CCCC(NC(c3cccc(Br)c3F)=O)C2)cc(C)n1 c1(C(=O)NCC#CCNC(C(C2CCOC2)OCC)=O)cc(OC)ccn1 c1(N(C)C(=O)OC(C)(C)C)ccc(NNC(=O)C2CCC(C#N)C2)cc1 N1(C(CC(C)F)=O)CC2CCCC(CNC(c3ccnc4c3CCO4)=O)C2C1 N1(C(CN(C(CSCCN(CC)CC)=O)CC)=O)CCSC2CCCC12 CC(C)C(C)S(=O)(=O)N=c1cc[nH]c(-c2ccccc2Cl)c1 N1(C(C23CCN(C(c4cncc(F)c4)=O)CC2C3)=O)CCc2cc(O)ccc2C1 N1(C(CC2(C)CC2(F)Cl)=O)CCN(C(=O)COC2CCOC2)C(CCO)C1 Cc1cc(C(N2CC(NC(C3CC4(C3)CC4F)=O)C(n3ccnn3)C2)=O)c(C)o1 C1(CNCCCS(CC)(=O)=O)(OC)CCOC(C)(C)C1 O=C1CCc2cccc(C(=O)NCC3CCCN3C(=O)C(=O)NCC(F)F)c2N1 c1(OCCC)ccc(C(=O)NCC2CC(NC(C3CC3C)=O)CC2O)c(OC)c1 c1(C(=O)NCCC(C)NC(c2cc(CC(C)C)[nH]n2)=O)c(C#N)cnn1C c1(CC(=O)NCc2cocc2C(N2CCC(c3cnn[nH]3)C2)=O)ccc(O)nc1 C1(O)(CNC(c2nn(CC)c(=O)cc2)=O)CCCN(C(=O)C(C(C)O)N(C)C)CC1 Clc1cccc(OC)c1.C12(CCOCC1)n1cc(nn1)CC1(CC1)CN2.C1CC1 N1(C(c2ncc(C)c(C)c2)=O)CC2CCC(C1)C2CNC(=O)Cc1cncs1 c1(C(N2CC(CCNC(c3c(C)nc(O)cc3)=O)C2)=O)c([N+](=O)[O-])cnn1C C(=O)(C(CC(F)F)NC(c1nccc(C)c1N)=O)NC(C(=O)OC)CC1CC1 CC(C)CC(C)CC(C)C(=O)NCc1cncc(-c2cn(C3(C(=O)O)CC3)nn2)c1 C=C1CC(C)(C(=O)N(CCCCN(C)C(c2cnoc2C)=O)C)C1 c1(CN2CC(CNC(c3ncc(C)s3)=O)OCC2)c(O)cc(Br)cc1F CC1CCCC(OCC(N2CC(CNC(c3cc(=O)cc[nH]3)=O)C2)=O)C1 Cc1noc(C)c1CN(C)C(C1CC(CCNC(C2CC2Cl)=O)C1)=O c1(OC)cccc(F)c1CC(=O)NCC#CCNC(c1ccc(=O)n(C)c1)=O C(=O)(CCC(F)(F)F)NCCN(C1CCCCCC1)C(C1C(C)(CC)C1)=O C1(N(C(C2CCOC2(C)C)C(=O)NC(CC)(C)C)C)CCc2nc(C)cn2C1 N1(C(CCCNC(C2CCC(C#N)CC2)=O)=O)C2CCC1CC(CO)C2 C1(C(N(CC(C(=O)OC)C)C)=O)CCN(C(C2CC3CCCC3C2)=O)CC1C C1(C(N(C)Cc2cncn2C)=O)CCC2(CC2)N1C(=O)C#CC1CC1 c1(C(=O)OCc2cn3cc(C)nc3s2)cnc2c(ccn2C)c1 CCCCCCCCCCCCCCC(=O)N1CC2CCC1C(CNC(C)=O)C2 C12(C(=O)NC3C(NC(c4ccc(CSC)o4)=O)CCC3)CC1CNC2=O Cc1ccc(C(N2CC3CC(NC(c4sc(O)nc4C)=O)C2C3)=O)cc1C#N C(CC(C)C(=O)NC(CNC(c1c(C)[nH][nH]c1=N)=O)CC)=CC c1(CC)c(C(N2CCC2CNC(C2CC=CCO2)=O)=O)cnn1CC(C)C S(=O)(=O)(c1c[nH]c2nc(F)ccc12)N1CCN(CC2S(=O)(=O)CCC2)CC1 C1(NC(C2CC(C)N(C)C2)=O)CN(C(C2CCSCC2)=O)CCC12CCC2 c1(CNC(c2n(CC)nnn2)C2(COC)CCOC2)ncc(F)cc1F Cc1cccnc1CCCNC1CCCC(CO)C1 C#Cc1cc(C(N2CC(NC(=O)C(C)(C)OCC)C(C)C2)=O)cc(Br)c1 N1(C(C2C(=C)C2)=O)CC2CC2(CNC(c2c(-c3ccccc3)noc2CC)=O)C1 Cc1ccccc1C=CC(=O)NCC(C)C(=O)N1CCCC1C(C)(C)C C(=O)(C(CC(C)C)NC(=O)CNC(=O)CNC(=O)C(C)(C)C1CC1)OCC c1(C(=O)OC)nc(C(=O)NCC2CC2NC(=O)Cc2csc(C)n2)cs1 c1(CC(=O)Nc2c(C(N3CCC(=C)CC3)=O)scc2)ccc(F)cc1Br C1(NC(c2c(C)scc2)=O)CCC(C)(CNC(C2CC2C2CC2)=O)CC1 Cc1ccc(COCC(C)C)c(NC(=O)NC2CC(=O)N(C)C2=O)c1 C(C1=NOC2CC12)(c1nnnn1C(C)(C)CC)NCc1cccc(COCC)c1 CC(C)(C)C(C)(C)C(=O)N1CCCC(NC(=O)CN2CCCNC2=O)C1 Cn1ccc2cc(NC(=O)NCC(c3ccc(O)cc3)O)ccc2c1=O Cc1cc(C(=O)NCC2CCCCN(C(=O)CC3C=CCC3)C2)c(C)c(C)c1 C1(c2n(CCCCC)nc(-c3cccnc3OC)n2)CCCC(=O)CC1 C#Cc1ccc(F)c(C(=O)NCC2CC2CNC(c2cncc3nc[nH]c23)=O)c1 C=CCC(CNC(=O)CNc1ccccn1)C(=O)N(CCCCC)CCO N1(C(c2ccc(=N)[nH]c2)=O)CCC(C2CN(C(=O)C3=NNC(=O)CC3)C2)C1 C#CCCCC(=O)NCC(C)(O)C(=O)N(C)C[Si](C)(C)C c1(C(=O)NC2(CC=C)CCN(C(C3CC(C)(O)C3)=O)C2)ccc(OCC)cc1Cl c1(C(=O)NC2C(NC(CCCOC)=O)CS(=O)(=O)C2)nn(C)c2c1CCCC2 C1(C)(CNC(CCc2onc(CC)n2)=O)CCN(C(=O)COC2CCCCC2)C1 C(=O)(C1c2c[nH]nc2CN1C(=O)CN1CC(C)(OC)C1)N1CC2C(CC)(C2)C1 C(CCCOC)(C(=O)N(Cc1ccc(C)o1)NC=O)OCC C(=O)(C(C(C)C)C(C)C)N1CC(C)(C(N2CC(C)CC(OC)C2)=O)C1 O=C(CCC(=O)c1ccc(Cl)s1)NC1CC(NC(C2CCC2)=O)C(O)C1 CC(C)CC(C)CN=c1nc(N(CCC(F)(F)F)C)c2c([nH]1)COC2 CCC(CNC(=O)Nc1cccnc1-n1cccn1)C(C)C n1(C(C)C)cc(C(=O)NCC(C)(C2CCC2)NC(c2cnc(C(N)=O)s2)=O)nn1 Cc1ccccc1CCC(=O)NCC1(C(C)(C)O)CN(C(=O)C(F)F)C1 N1(C(CC(CC)C(C)C)=O)CCOC2(CCCN(C(C3CCc4cncn4C3)=O)C2)C1 C(C(C)(COC)C(=O)NC(C)Cc1cn(Cc2nc(C(=O)O)cs2)nn1)OC N1(C(C(CNC(=O)C=C(C)CC2CCC2)OC2CC2)=O)CCN(CC)CC1 C(=O)(CC(CN(C)C)C(F)F)NCC(CNC(CC1(C=C)CCOCC1)=O)(C)C N1(C(c2c(Cl)cn(CC)n2)=O)CCc2ccccc2C(NC(=O)C2CC2)C1 N1(C(c2ccc(C#C)cc2)=O)CCC2(CC(NC(=O)Cc3cc(C)ns3)CO2)C1 C1(C(=O)NC(C)CC2CN(C(c3cn(C(C)(C)C)cn3)=O)C2)CCCCC1O C1(CCNC(C=CC=CC)=O)C(C)CCCN1C(c1cc(CN(C)C)on1)=O Cc1cc(C(N2CCC(CCC(N3CC(C)CC(O)C3)=O)CC2)=O)c(C)n1C N1(C(c2cccc(Br)c2C)(CCCCCC)C(=O)NC)CCc2oc(C)nc2C1 C=CC1(C(=O)NCCOC(C)(C)CNC(=O)C(F)C(F)(F)F)CCCCC1 C(CCSC)(C(=O)NC1CCCN(C(c2n[nH]cc2Br)=O)C1)OC N1(C(Cc2nnc(C)o2)=O)CCC2CCN(C(=O)C(n3ccnc3C)C)CC12 C1(CC)CCCC1(C)C(=O)N(CC(C)(C)CNC(c1ccc(C(F)F)cc1)=O)C c1(C(=O)NCC(c2ccsc2)O)ccc(C2CC2(F)F)cc1 c1(C(=O)NCCCOCCCC)coc2c1CN(C(=O)C(C1CCOCC1)F)C2 N1(C(c2c(CC)n(C)nn2)=O)CCN(C(=O)CCc2cnn[nH]2)CC1CC1CC1 Fc1ncccc1OCC(N(C1CCC1)CCOCC(C1CCCCO1)=O)OC C(C)(N=c1nc(Cl)[nH]c(C)c1C#N)C1CCC(NC(CCC)=O)CC1 c1(C(N2CC(C3(NC(C(C)OCC4CC4)=O)CC3)C2)=O)cn(C)c2ccccc12 c1(C(=O)NC23CN(C(CN(CC)CC)=O)C(CC2)C3)cc(C)c(F)cc1F CCCCCC(CC)C(=O)NC(CN(C(=O)Cc1ccsn1)C)CC c1(C(=O)NCCCN(C(=O)C=CC(F)(F)F)C(C)C)ccc2ncnn2n1 c1(C(N(C(C(=O)NC(c2cnnn2C)C)C)C)=O)ccc(C2CC2)cc1 c1(SC)ccc(Cl)c(C(=O)NCC2(CNC(C3(C#N)CC3)=O)CC2(F)F)c1 N12C(CC3COCC13)CNC2=O.N(C1CC1)CC.C(C)=O C(=O)(CCCC(F)F)NC12C(CN(C(C3CN(CC)C(=O)C3)=O)C1)C2 c1(CS(=O)(=O)NC(c2ccc(F)cc2)C)ccc(Br)cc1F CC1CC2(CC(C(=O)NCCCCC(N3CC(C)OC(C)C3)=O)C2)C1 N1(C(Cc2cc(C)ncc2)=O)CCC(O)(C(C)NC(=O)CC2CCOC2)CC1 c1(OC)cc(Br)cc(NC(N2CCN(C3CC3)CC2)=O)c1OC C1(C(N2CC(O)(CNC(c3cc4[nH]ccc4s3)=O)C2)=O)CC2(CCOC2)C1 C1(CC)(CC)NC(=O)N(CC(=O)NCC2CN(C(=O)C(C)NC(N)=O)CC2O)C1=O Cc1[nH]nc2ccc(C(N3CC(C)(NC(=O)CC(C4CC4)C4CC4)C3)=O)cc12 N1(C(Cc2cn(C)nc2)=O)C2CCCC1CN(C(c1ccnc3ccnn13)=O)C2 n1(CCC)ncc(C(=O)NCC2(NC(=O)C(O)C3CC3)CCCCC2)c1Cl c1(C(=O)NCC(CN(C(CC(C)N(C)C)=O)C)O)cc(F)c(Cl)cc1F c1(C(N(CC(C(=O)NCc2csc(C)c2C)C)C)=O)coc2c1COC2 N1(c2nccc(=NCCNC(C3C(OC)C3)=O)[nH]2)CCc2cccc(CO)c2C1 N1(C(CCCCC)=O)CC2CCCC2(CNC(=O)C2=COCCC2)C1 CCC(CC)CC(F)C(=O)NC12CC(NC(c3cn(CCO)nn3)=O)(C1)C2 c1(N2CCCC(CC(C)C)C2)cccc(S(=O)(=O)N(CCCF)C)n1 C(=O)(C(C)(Cl)Cl)N1CC(N(C)C(C2(NC(=O)OC(C)(C)C)CC2C(F)(F)F)=O)C1 C1(NC(C(C)(C)N(S(C)(=O)=O)C)=O)CN(C(c2c(C(F)(F)F)coc2C)=O)CC1O N1(C(c2ccc(OCC)cc2)=O)CCCN(C(c2ccon2)=O)C(CO)C1 n1(CC(=O)NC(C2CCCC2)CNC(C(C)NC(C)=O)=O)cnc2c1CCCC2 c1(C(=O)NCC(C)NC(c2ncc(OC)cn2)=O)c[nH]c(C)c(Cl)c1=O N1(C(CC(C)C)=O)CC(CNC(c2cccc3sccc23)=O)CC12CCOCC2 C1(NC(C2CC(OCC)C2)=O)CN(C(=O)CCCC(C)=O)C2(CCOCC2)C1 N1(C(C=COCC)=O)C2CCC1CC(CNC(=O)CC1COC(C)(C)CO1)C2 CCCCC(C(=O)NC(c1nn[nH]n1)CC)NC(c1cc(C#N)n(C)n1)=O CCCCCC(CC)C(=O)NCC1(NC(=O)CCNC(C2CCC2)=O)CCCC1 c1(CC2(C(=O)NCC(CNC(=O)Cc3ccon3)OC)CCC2)cccc(Cl)c1 CC1CC(C)N(C(=O)CSS(C)(=O)=O)CCN1C(=O)Cc1cc[nH]n1 c1(C(N(C2CCN(C(CC3CN(C)CC3O)=O)C2)C)=O)ccnc2c1CCO2 c1(C(N2CCC(N(C(C3CC3F)=O)CC)C2)=O)cc2cc(Br)cnc2s1 C(CS(=O)(=O)N(C1CCC1)Cc1cnn(C)c1)(C1CC1)OCC C1(C(N(C(C)CN(C)C(c2ncc(F)cn2)=O)C)=O)CCCC(=O)N1C c12ccc(cc1)C(=O)NCC2SC.c1(NC(=O)C(O)C(C)C)ccccc1CO c1(C(=O)NC(c2cccc(C)c2)C(C)(C)C)ccc(Cl)c(Cl)c1 c1(C(N2C(CNC(C3C(OCC)C3)=O)CC2)=O)cc(OC)c(O)c(C2CC2)c1 CCCC(CC(=O)N1CCCC1C(=O)OC)NC(=O)C(O)Cn1cncn1 C1(n2cc(-c3ccc(OC)cc3)nn2)CON(C(=O)C(C)n2cc(Br)cn2)C1 Cc1ccc(CN2CCC(C(N3CCN(C(C)C)CC3)=O)C2)cn1 CC(C)(C)CCC(=O)N1CC2C(C(N3CCOC(C(C)(C)C)C3)=O)C2C1 C1(F)(C(N)=O)CCN(CC(=O)Nc2cccc(OC(F)(F)Cl)c2)CC1 C(=O)(C1=CCCSC1)NCC1(F)CCN(C(c2scc(C(=O)OC)c2)=O)C1 CC1CC2CN(C(=O)C3=CC(O)C(NC(=O)C=C4CCOCC4)C3)CC12 c1(CC(=O)N(C(C#C)C2CCC2)CC)csc(N(C2CCCO2)C)n1 c1(C(N(C2CCN(C(C(CCC)C#N)=O)C2)C)=O)cc(S(N)(=O)=O)ccc1F c1(C(=O)NCC(C)(CO)NC(c2ccnc(CO)c2)=O)ccn2nnnc2c1 N1(C(c2sc(C)c(Br)c2C)=O)CC2CN(C)C(CO)C2C1 O=C(CCCNC(c1ccncc1)=O)NC1C=CC(CNC(c2cn[nH]c2)=O)C1 C1(C(N2C(CN(C(C=CC(=O)OC)=O)C)CCCC2)=O)CCc2c(n[nH]c2C)C1 O=C1CCCN(C(C2C3CC2N(C(C2CC4(CSC4)C2)=O)C3)=O)C1CCO N1(C(C2(NC(CC)=O)CCCC2)=O)CC(n2cc(C(C)O)nn2)C(C)C1 c1(C(=O)NC2(CO)CCCN(C(C(CC)COC)=O)C2)cc(F)c(F)cc1Cl N1(C(C(CC(N)=O)O)=O)CC(O)(C2(CNC(=O)CCn3ccnn3)CC2)C1 CC(CC(=O)NC1CC2CC(C1)N(C(=O)CSc1cnn(C)c1)C2)CC(F)(F)F c1(CC(=O)NC2CC3CC2N(C(C2CC2C2CCC2)=O)C3)cc(F)cc(Cl)c1 N1(C(C(C)OC2CCCC2)=O)CCC(CNC(c2ccnn2C(C)(C)C)=O)CC1 c1(C(=O)NC(C(=O)OCC)CN(C)C)ccc(=O)n(-c2ccc(F)cc2)c1 Cc1ccc(F)c(-c2cn(CCC(=O)NC3(C)CCCCC3C)nn2)n1 CN(C)S(=O)(=O)NCC(=O)NC1CC(NC(C2CC3(CC3)CO2)=O)C1 c1(NC(C(=O)NCCOC2(C)CCCC2)=O)ccc(SC2CC2)cc1 CCCC(O)CC(=O)NCC1(NC(c2cc(Cl)c(Cl)s2)=O)CCOCC1 CC(C)CC(C#N)C(=O)N1CC(NC(C23CCC(N(C)C)(CC2)C3)=O)C2(CC2)C1 C1(CC(N2C3(C(N(CCNC(C)=O)C)=O)CC(C2)C3)=O)CCN(OC)CC1 C=CC(C)(CCOC)C(=O)NCCN(C(=O)COCc1nnc(C)s1)CCC CC1c2c[nH]nc2CCC1C(=O)NC1CCN(C(=O)C(F)(F)CN(C)C)CC1O c1(C(=O)NC(CCCC)CNC(C2(OC)CCC2)=O)cc(Cl)c(OC)cc1C C(=O)(C(O)C(C)(C)C)NCC1N(C(c2ccc(-c3nc(C)sc3)s2)=O)CC1 C1(CCC2N(C(CCSCC)=O)CCC2)CCN(C(C2CC3CC2C3)=O)CC1 CC(N=c1ccc([N+](=O)[O-])c(O)[nH]1)C1CN(C(=O)CC2COC(=O)C2)CCO1 c1(C(N(C)CC2CCN(C(C=C(C)C(F)F)=O)C2)=O)cc2cccnc2o1 CC1CC(NC(=O)CO)CCN1C(c1ccc(Cc2nc[nH]n2)cc1)=O C1(CC)CN(C(c2ccsc2)=O)CCC1NC(c1cnc(C)cc1Cl)=O c1(CC(=O)NC2CC3CC(NC(C(CC)C)=O)C2C3)cc(F)c(F)cc1F Cn1cc(C(N2CC3CC(NC(=O)CC4CC4(Cl)Cl)C2C3)=O)n2cncc2c1=O CCC(CC(F)(F)F)C(=O)N(C(C)CN(C(=O)CCN(CC(F)(F)F)C)C)C c1(C(=O)O)ccc(O)c(CNCC2CCCCN2C(c2cn(C3CC3)cn2)=O)c1 N1(C(=O)CCCC2CCCCC2=O)Cc2ncsc2C1 c1(OCC)nc(C)ccc1C(=O)NCC1CCCN1C(c1ncsc1NC)=O C1(C(N2CC(NC(CCc3ccc(C)nc3)=O)(CO)C2)=O)CCCCC1C1CC1 c1(C(=O)NC2(CO)CCN(C(=O)COc3ccsn3)C2)cn2ccc(CO)cc2n1 N1(C(C2(C)CC3CC3C2)=O)C2CCCC1CN(C(c1sccc1F)=O)CC2 C(=O)(C(O)CC(C)C)N1C(C(C(=O)NC(CC=C)C(=O)OCC)(C)C)CCC1 C(=O)(CC(=O)NC(CNC(=O)CC1CC=CCC1)CO)OCCC(C)C N1(C(c2cn(C)nc2)=O)CCC(C)(C)C(C(=O)NCc2cnc(O)c(F)c2)C1 c1(-n2cc(C3CCCN(C(c4[nH]ccc4C4CC4)=O)C3)nn2)ccccc1[N+](=O)[O-] C1(COC)(NC(=O)C(n2ccnc2C)C)CN(C(=O)CN(C)C(C)C)C1 c1(C(C)=O)ccc(C(=O)N2C3CC2C3)nn1.C1(C(=O)N(C)C)CC1C(N)=O c1(C(=O)NC2CC(CN(C)C)C2)ccc(-n2ccnc2)cc1 c1(C(=O)NC2CN(C(C(C(=C)C)(C)C)=O)CC2O)cc2nc(Cl)ccc2s1 Cc1nc(C#N)c(COCCC(=O)N(CC(C)NC(=O)Cc2ncc(C)o2)C)o1 c1(CC(=O)NC2CN(C(c3cnc(O)s3)=O)CC23CC3)ccc(Cl)c(Cl)c1 C1(C(N2CC(CCC)OCC2)=O)C2CCN(C(=O)C(C)OCC3CC3)CC12 CC(C(=O)N1CC=CC1(C)C(N1CCCN(C2CC2)CC1)=O)S(N)(=O)=O C1(NC(C2CC(O)C2)=O)CC2(C(=O)NCCOC3CCC3)COC1C2 c1(C(=O)OC)cccnc1C(N1CC2CC2(NC(C2CC(OC(F)(F)F)C2)=O)C1)=O C1(C(=O)NC2(CNC(CCN(C)CCO)=O)CC2)CC2(C1)CC21CCC1 CC1CN(C(c2cnn(C)c2)=O)CC1NC(c1cnc(O)n1C)=O C(CCN(C)C(C1(n2cccn2)CCC1)=O)(C(C)C)NC(C(C)NC(CC)=O)=O C(=O)(C1=C(Cl)CCC1)N1CC(C(C)NC(=O)C(Cl)=CCl)OCC1 N1(C(C(C)NC(=O)OC(C)(C)C)=O)CCCC(O)(C(=O)N(C2CCCC2)C)CC1 N1(C(CCC#C)=O)CCC(C)C(NC(c2ccc(OCCO)cc2)=O)C1 c1(C(N2CCC(F)(CNC(C3CC(OC)(OC)C3)=O)C2)=O)ccc2ccoc2c1 N1(C(C(CN(C)C)(C)C)=O)CC(CNC(C2C3CCCCC23)=O)C2(CCC2)C1 c1(C(C(N2CCCC(C(=O)OC(C)(C)C)C2)=O)NC)cc(F)ccc1F N1(C(COCCCCC)=O)CCC(C(C)(C)C)(CNC(c2cn(CC)nn2)=O)C1 C1(CCOC)CN(C(=O)C(=Cc2ccco2)C)CCN1C(=O)CCC1CCCO1 N1(C(CN2CC(=O)NCC2)=O)CC2CCN(C(C3(Cl)CC3(F)F)=O)CC12 C(=O)(CCP(C)(C)=O)NC(C)CC1CCN(C(=O)COCC(F)(F)F)CC1 c1(C(N(CC(=O)NCC(CC)O)C(C)C)=O)cc(C(C)=O)c[nH]1 C1(C(=O)NCc2ccc(OC)c(O)c2)CN(C(=O)C(C)(O)C(C)C)CCC1(F)F C1(NC(c2c(CC)csc2)=O)CC(F)CN(C(=O)C(Br)=C(C)C)C1 C1(NC(c2cc(OCC)c(OC(F)F)cc2)=O)Cc2ccc(C#N)cc2C1 C(CCCC(C)NC(=O)C(CCC)OCC)NC(C1(C#C)CC1)=O CC1CC(c2cccnc2)N(C(C2CCCN(CCC(C)(C)C)C2)=O)C1 N1(C(C(CC)N(C)C)=O)CC2CCN(C(c3cn[nH]c3)=O)C2C1 C[S+](C)CCC(O)C(=O)NC12CC(NC(=O)CC3SC(=N)NC3=O)(C1)C2 c1(C(C(N2CCC(N(C(c3c(CC)ncs3)=O)C)C2)=O)(C)C)ccc(OC)cc1 CCC(C(=O)NCC(C1CCC1CN)=O)NC(=O)C1CC1 C1(C(=O)NCC(NOC)=O)CC(F)CCN1C(C1CC(O)CN1C)=O C(=O)(N1CCC(C(N2CCOC(C)(C)C2)=O)O1)C1C(C)=CCS1 C1(CNC(COC2CCCC(C)C2)=O)N(C(=O)CCC2CC2)CCCC1(C)C c1(SCC(=O)NCCC2(NC(CCCC#C)=O)CC2)ccc(F)c(F)c1 N1(C(=O)Nc2c3cnn(CCOC)c3ncn2)CCOC2(CCSC2)C1 C#CC1(C(=O)Nc2cccc(C)c2Br)CCN(C(=O)C(=O)NCCOC)CC1 c1(C(C)NC(N2CC(C=C)(CC(=O)OC(C)(C)C)C2)=O)ccc2nc(O)[nH]c2c1 c1(CN2C(C(N3CCOCC3C)=O)CC(=C)C2)c(F)cc(C)cc1F C1(NC(C2CCN(C(C)=O)C2)=O)CN(C(=O)COCCF)CC1O C1(NC(N2CCN(c3nccc(OC(C)(C)C)c3)CC2)=O)OCCC1CC(O)C c1(OC)nccc2c1CN(C1CC(C(N)=O)C1)CC2 CC(C)(CO)C(=O)NCCN(C(c1cc(-c2ccccc2)[nH]n1)=O)C1CC1 c1(C(=O)NC2CC(C)(NC(CC3(OC)CC3)=O)C2)cccc(-c2noc(C)n2)c1 c1(C(N2CC(OC)(CNC(c3ccccc3C(C)C)=O)C2)=O)c(C)cncc1C N1(C(COCCC#N)=O)CCc2ccc(C(=O)NCC3CCCCO3)nc2C1 N1(SC(Sc2n(C3CCN(C)CC3)ccn2)=S)CCOC2(CCC2)C1 c1(C(=O)NC(C2CC=CCC2)C(=O)NC2CCN(C(=O)OC)C2)nnn(C)c1N c1(CNC(C(CC2CCOCC2)NC(c2ccc(CO)s2)=O)=O)cc(=O)cc[nH]1 c1(C(N2CCC(OCCNC(c3ccc(F)c(Cl)c3)=O)C2)=O)ncnc(O)c1F N1(C(C(C(C)C)n2cncn2)=O)CCN(C(c2ccc(C#N)[nH]2)=O)CC1CF c1(-c2cn(CCc3cccc(C(=O)OCC)n3)nn2)cccc([N+](=O)[O-])c1 C(=O)(C(O)C(C)(C)C)N1CC(CC(C)NC(C=Cc2nnc(C(C)C)o2)=O)C1 C1(NC(CC(C)OC)=O)COC2(CCN(C(=O)C(F)=C3CCC3)CC2)C1 C(C(=O)N(C1CCN(C(c2nocc2-c2ccccc2)=O)C1)C)(C(C)C)OCC Cc1nn(C)c(C)c1OC(=O)CSCC(=O)NCCNC(=O)CC1(C)CCC1 N1(C(C23C(CN(C(c4ccncc4Cl)=O)C2)CC3)=O)CCC(CO)C(F)(F)C1 Cc1cc(C(=O)NC(C(=O)NC2CC3(CC3)C2)c2ccoc2)ccn1 c1(CCCC(=O)NC2CC(NC(=O)C(F)(F)C3CCCC3)C2)cc(F)ccc1F N1(C(=O)NCC2C(OC)CCCC2)C2CCC(O)C1CCC2O S(=O)(=O)(c1cc(Cl)sc1C(=O)NC1CC(C)N(C(=O)CCCC2CC2)C1)NC N1(c2ccc(C(N(C)C)=O)cc2)CC2CC(NC(=O)CCCCCBr)CC2C1 c1(C(=O)NC23C(CN(C(Cc4ccc(OCC)cn4)=O)C2)C3)cnc(O)c(C)c1 c1(C(=O)NC2CCN(C(c3cnc(OCC)s3)=O)C2)ccc(Cl)cc1[N+](=O)[O-] c1(C(N2C(CNC(CC(=C)C)=O)CC(OC)C2)=O)cnn2c(=O)cc[nH]c12 CCCC(C)C(=O)N1CCCC(CNC(=O)Cn2nc(C(F)(F)F)cc2Cl)C1 c1(OC)cc(C(N2CCC3(NC(=O)CNC=O)CCCC23)=O)cc(Br)c1OC C1(C(=O)NC2CCN(c3nc(OC(C)C)c(F)cn3)CC2)CCCCC(F)(F)C1 N1(C(CCCC(=O)NCC)=O)CC2=C(C1)CN(C(=O)C(C)(O)CC(C)C)C2 C1(C(=O)NCc2c(C)noc2C)CC(C)CN(C(=O)CSc2ccccc2Cl)C1 c1(NC(=O)NCC=C)ccc(C(=O)N(CC(C)CNC(=O)CS(=O)CC)C)cc1 C12(C(=O)NCC3(C)CCC(NC(C4CC(O)C4)=O)C3)CCCN(CCC1)C2 c1(C(=O)NC(CC(C)NC(c2c(CC)c(C)sc2)=O)C)cccc([N+](=O)[O-])c1 C(=O)(C1=CCCC1C)N(CCC(=O)NCC(=O)NCCC)C1CCC1 C1(C(=O)NC2(CNC(c3c(C)n(CCO)cc3)=O)CCOC2)COCC(C)(C)O1 C(=O)(C(O)CC[S+](C)C)N(C(C)C)CCN(C)C(C1(C#N)CCSCC1)=O CP(C)(=O)C1CCCCC1C(=O)N(CCNC(=O)Cc1cncnc1)C1CC1 Cc1cnn(C)c1CC(=O)NC1CC(C(=O)N(C)CCC2CC2)C1(C)C c1(OC)ccc(C(=O)NC2CC2NC(=O)CC2(C)CCCC2)c(Br)c1 N1(C(CC(CC)C(C)(C)C)=O)CCC2(CC1)CN(C(=O)CCC(N)=O)CC2CO c1(C(=O)NCCCC(C=C)(C)C)cc(OC)c(N)cc1F N1(C(C2C(C)(C)CCO2)=O)CCC(C(=O)NCC2(C)CCCS2)=C(F)C1 C1(CNC(=O)C(O)c2ccco2)CC2CCC1N(C(C1COCCO1)=O)C2 CCC(C)C(C(=O)NCC1C2CCCC12)N(C)C(C1CS(=O)(=O)C1)=O c1(C(=O)NCC(C)N(C(=O)C(C2CCOCC2)C)CC)cc2cccnc2[nH]1 C=CC(C)(C)CC(=O)NC1CC(OC)CN(C(=O)CN2CCCC2CO)C1 c1(C(=O)NCC(CNC(C=CCC)=O)CO)cn(C)nc1Br c1(OC)ccc2cc(C(=O)NC3CC3NC(C3CC(=O)N(C)C3)=O)c(C)nc2c1 N1(C(c2cc(COC)no2)=O)CC(NC(C2CCS2(=O)=O)=O)CCC1C C1(NC(C=CC2(C)COC2)=O)CCCCN(C(=O)CC2CNC(=O)C2)C1 c1(CC)ncsc1C(=O)NC(C(=O)N(C)CC1CCOCC1)C1CCOC1 C1(C(=O)NC(CO)C(C)NC(=O)CSc2ccccc2)(OC)CCOC1 Cc1cc(C(=O)NCC(CNC(=O)C(O)c2ccsc2)CO)n(C)n1 N1(C(C(C)NC(=O)NC)=O)CC2CCN(C(=O)C=Cc3ccncn3)CCC2C1 c1(OC)ncnc(C)c1C(=O)NC1COCCN(C(C2(O)CCC2)=O)C1 C(=O)(N=c1[nH]sc2ncccc12)C1CCN(C(c2ccc(C)c(CO)c2)=O)C1 O=C(CCCCC(F)F)NCCC1CCCCN1C(c1cc2sccc2cn1)=O N1(C(CSCCC(C)C)=O)CCOCC1CC(N1CCCCC1CO)=O CC1CCCN(C(C)C(=O)NCCn2cc(CC(C)(C)O)nn2)C1 C1(CCC)CC1N=c1[nH]c(N(C)CCOCCN(C)C)nc2c1CC(C)CC2 C1(NC(CCSc2nc(C)[nH]n2)=O)CCN(C(=O)CC=C(Cl)Cl)CC12CCC2 N1(C(C(CNC(c2cscc2Cl)=O)O)=O)CC2CCCC(O)C2C1 N1(C(C(C)SCCCC)=O)CC(C2CCCCN(C(=O)COCC3CCC3)C2)C1 Cn1ncc(C(=O)NCC(F)(F)Oc2ccc(F)cc2)c1N CC1(CNC(C2(CF)COC2)=O)CC(F)(F)CN1C(=O)Cc1nc([N+](=O)[O-])n[nH]1 c1(C(N(CCNC(C2CCC(C)S2)=O)C2CC2)=O)ccc(N)c2c1CCCC2 CCCCC(C(=O)NCCCNC(=O)CCCc1ccc(O)c(F)c1)NC(N)=O c1(C(=O)NCC2C=CC(NC(C(C)=C(CC)C)=O)C2)ccc(C#N)[nH]1 C1(c2nnnn2CC(F)F)(NCCC(=O)NC)CN(C)CC1C N1(C(C(C)NC(CC)(C)C)=O)CC(NC(=O)CC2(C)CCC2)CC2(CC2)C1 c1(-c2cc(C(N3CCN(CCOC)CC3)=O)ncc2)cc(OC)cc(C)c1 C1(C(=O)NC(C2CCN(C(CC(C)(F)F)=O)CC2)(C)C)CCC12CCOCC2 C=C(C)C(CC(=O)N(CC(=O)NCc1ccc(C)cc1C)C1CC1)OCC c1(CC(N2CC3C(NC(CNC(CN(C)C)=O)=O)C3C2)=O)cc(F)c(F)cc1F CC(=O)CCCC(=O)N1CC(F)CC1CC(N1CCC(CN(C)C)CC1)=O c1(CC(=O)NC2C(NC(c3c(OC)cc(CO)cc3)=O)C2)cccc([N+](=O)[O-])c1 C(CC(C(=O)NCc1nc[nH]n1)NC(C1CCCCN1C)=O)OCC C(=O)(CCN1C(=O)NCc2ccccc21)NC(c1c(C)n(C)nc1)C(=O)O N1(C(CCc2cc(C)[nH]n2)=O)CCC(NC(=O)CN2CC(C)(C)C2)C1(C)C N1(C(=O)CCCF)CCCCC(C2CN(C(c3ccc4ccsc4c3)=O)C2)C1 N1(C(C2C(OCC)C2C)=O)CC=C(CNC(=O)CCc2nc(C)no2)CC1 CCC(C)(COC)C(=O)N1CCCC(CCCCNC(=O)CN2CC3CC3C2)C1 c1(OC)ccc2nccc(C(N3CC4CN(C(c5ccc[nH]5)=O)CC4C3)=O)c2c1 C(=O)(CCCCC#N)NC(c1ccccc1)CNC(CCSc1n(C)nnn1)=O c1(N2CCN(C(C(C)C)=O)CC2)nc2c(c(=NC3CSC3)[nH]1)COC2 N1(C(CC2(C=C)CC2)=O)CC2CC2(CNC(c2ccnc(C(F)F)c2)=O)C1 CN1CC2(CCCN(C(=O)C(N3CCC4C(C3)C4(F)F)=O)C2)CC1=O c1(C(=O)NCC(C2CC2)NC(C2(C)CC2(Cl)Cl)=O)cccc2c1OCCN2 C1(CC(N2C(Cc3cn(CCC(=O)OC)nn3)CCC2)=O)CCCC(C)(C)O1 C1(SC)CN(C(C2CC(C)C2)=O)CC1NC(C1(n2cccn2)CCC1)=O Cc1ccc(F)c(C(=O)NCC(C(C)C)NC(=O)CC2C(C)C2(F)F)c1 N1(C(c2ncc(C)nc2)=O)CCC(CNC(=O)C(O)c2ccco2)C(C)C1 C=CC(C)(O)C(=O)NCC(CC)NC(=O)Cn1cc(C2CC2)cn1 N1(C(=O)CSC2CCCCO2)CCC(O)(NC(C23CCCC2C3(F)F)=O)CC1 Cc1nnc(CN2CCC2C(=O)NCc2ccn(CCF)n2)o1 C1(NC(C2(NC(CN(CCOC)C)=O)CCC2)=O)CCCC12CC2 N1(C(C)C)C(=O)COCC1C(=O)NC1CC(F)(CNC(C2CC=CC2)=O)C1 c1(C(c2nnnn2C2CC(C(=O)OC)C2)NCCC(C=C)C)ccc(NC)nc1Cl C(C(=O)NCC1COC1)(C(C)(C)C)NC(CCOCCOCC)=O C1(CNC(C2CCC(C)C2)=O)CCC2CN(C(c3ncccc3O)=O)CC12 C(=O)(C(F)(F)CCn1ccnn1)NCC(CC)NC(c1nccc(C)c1O)=O Nc1c(F)ccc(Cl)c1C(=O)NCC1(CCNC(C2(F)CC=CCC2)=O)CC1 CC(C)CC(C(=O)NCC1(O)CN(C(C2(C)CCC(O)CC2)=O)C1)n1ccnc1 C(=O)(C(C)(C)CC(F)F)NCC(C)NC(C1(CC)CCC1)=O O=C(N=c1nc2cc(Cl)ccn2[nH]1)c1ccc(-c2ccc(O)c(I)c2)nn1 c1(C(N(C)CC2CCN(C(C3(OC)CC3)=O)C2)=O)ccc(C(F)F)c(F)c1 Cc1cc(C)c(C(=O)N(C2CN(C(c3ccncc3Cl)=O)C2)C)[nH]1 CCCCC(CC)C(=O)N1CCN(C(C2CCC(OC)CC2)=O)C(COC)C1 C1(C(=O)NC2CCCCCN(C(CCCC)=O)C2)CC(=O)c2cc(Cl)ccc2O1 N1(C(c2c(C)onc2)=O)CCC(C2CCCN(C(=O)CCn3cccc3)C2)CC1 c1(C(C#C)OC(C)CC)ccccc1 c1(CN(CCS(N)(=O)=O)C)nn(CC(F)(F)F)cc1Br c1(C(=O)OC)nc(C(=O)N(C2CC(NC(=O)C(CC3CC3)OC)C2)C)cs1 C1(C)(NC(CC2C(C)CCN(C(c3cc(SC)oc3)=O)C2)=O)CCCC(C)(C)C1 c1(C(N2CC(CC(C)NC(=O)CCC3CCC(=O)NC3)C2)=O)cccnc1S c1(NC(C(N2C(C)(C(=O)NC)CC2)c2csc(C(C)(C)C)c2)=O)ccccc1Cl C12(CC)CCC(C(=O)NC3CCN(C(C4CC5CCC4C5)=O)C3)(CC1)CO2 c1(CC)cccc(NC(c2cc(CNC(=O)C(CC(C)C)N(C)C)[nH]n2)=O)c1F c1(C(N(C)CC2(CNC(c3cc4sccc4s3)=O)CC2)=O)cncn(C)c1=O O(C1CCc2c(F)cc(F)cc21)C(c1ccc(C(F)(F)F)c(Br)c1)=O N1(C(c2c(CC)non2)=O)CCC(C(=O)Nc2cc(C)c(C)cc2C)C(C)(C)C1 c1(C(N(CCNC(C2CC(OC)C23CCC3)=O)C)=O)cc2c(C)ccc(F)c2[nH]1 CCC(C)CCCC(=O)NCC1CC1CNC(c1cc(N(C)C)ccn1)=O c1(CNC(CN(C2CC2)CC)=O)ccc(CCNC(=O)C(F)=C(C)C2CC2)cc1 c1(C(N(CC(C)N(C(C=CC)=O)C)C)=O)ccc(C)c(OC)c1 CC1C(C(=O)NCC(=O)N(C)O)CCN1C(=O)CCCCC1CC1 c1(OC)cnc(C(=O)NC2CCOCC2C(=O)NOCCCO)cn1 c1(C(=O)NC(C)(CNC(c2cnccn2)=O)CO)nc2c(s1)COCC2 c1(C(N2CCC(CN3CCCC3C(=O)N3CC(O)CO3)C2)C)ccc(OC)c(F)c1 N1(C(c2c(C)cn(C)n2)=O)CCC2CC1CN(C(=O)CCC1CCC(=O)NC1)C2 c1(CCC(=O)NC2CC3CC2N(C(c2n[nH]cc2F)=O)C3)nnc(S)nc1O c1(C(N2CC(C(=O)NC(CCOC)COC)(OC)C2)=O)cccc(C)c1C c1(C(=O)NC(C(C)NC(CCC=C(C)C)=O)CO)ccc(Br)c(F)c1F C(N=c1cc(C2CC2)nc[nH]1)C1(F)CC(NCCOc2ccc(C)c(C)c2)C1 n1(C(C)C)ccc(C(N2CCC2CNC(C2(C(F)F)CC2(F)F)=O)=O)n1 C(=O)(C(C)C(C)NC(c1cc(Cl)n(C)n1)=O)NCC(C1CC1)SC c1(OC)cccc(NC(=O)C(C)(C)C2CCCO2)c1N1CCN(C)CC1 c1(C(=O)NC2(CNC(CC(CCC)O)=O)CCCC2)cc2cnccc2o1 N1(C(C2(COC)COC2)=O)CCC2(CC2NC(=O)CC(=O)N(C)C)C1 N1(C(C(CC)C(C)C)=O)CCN(C(=O)CC2(OC)CCC2)CC(O)C1 c1(OC)cccnc1C(=O)NCC(C)(C)CNC(c1cn(CCF)nn1)=O CC1CN(C(c2ccnnc2O)=O)CC2(CCN(C(=O)CC3OCCO3)CC2)O1 Cc1cc(NC(C2(C)CCCN2Cc2ccc(F)nc2)=O)ccc1C#N CC1CCCN(C(=O)Cc2cccc(OC(F)F)c2)C1CNC(=O)COC1CC1 c1(CNC(C(CNC(=O)COC2CCCC2)N(C)C)=O)ccc(F)cc1F N1(C(CCC(=C)Cl)=O)CCCCC2(CCN(C(C34CCC(N=[N+]=[N-])C3C4)=O)C2)C1 c1(C(=O)NCCNC(CC2(C)CC2(F)F)=O)ccc(N)cc1C(F)(F)F C(C)(CCCCNC(c1ccc(F)cn1)=O)NC(CC(=C)Br)=O C1(CNC(c2n(C=C)ncc2)=O)C(O)C(O)CN1C(=O)C(c1c(C)n[nH]c1C)C CN1CCn2cc(C(N3CCCC3CN=c3[nH]nc(C(C)(C)C)s3)=O)nc2C1=O C(CCCC(=O)NCC1CCCN1C(c1cccnc1C1CC1)=O)OCC N1(C(C(C(=C)C)(C)C)=O)CCCCC12CN(C(=O)CC(=O)NCC)C2 C1(C(=O)NCC(CO)NC(c2c(C(C)C)noc2)=O)CCc2nccn2C1 Cc1cc(C(=O)NCC2COCCN2C(c2snnc2C)=O)cc(Br)c1 Cc1cc(C#N)ccc1C(N1CCN(C)CC1CNC(C1(F)CCOCC1)=O)=O C1(Nc2nc(OC)c(C)cn2)CCC2(C1)CN(C(=O)C(C)n1ccnc1)C2 C1(O)(CNC(C2CC(N(C)C)C2)=O)CCCN(C(c2ccc(Cl)c(N)c2)=O)CC1 c1(C(N2CCC(CNC(c3ccnc(C(F)(F)F)n3)=O)C2)=O)cc([N+](=O)[O-])c[nH]1 N1(C(c2cc(CC)n(C)n2)=O)CC2CCC(Nc3cncc(Cl)n3)CC2C1 C(=O)(CC(C)(C)c1ccc(F)cc1)OC(c1ncc(C)o1)C1CC1 Cc1cncc(C(=O)NC2CCC(F)(CNC(c3nc(Cl)c(Cl)s3)=O)C2)n1 N1(C(c2ccn(C(F)F)n2)=O)CCCN(S(=O)(=O)Cc2ccc(F)cc2)CC1 C=CCC(CC(C)C)C(=O)NC1CC1NC(c1ccc(C(F)(F)C(F)F)cn1)=O c1(OCC(=O)NC2CC(CNC(CC(CC)O)=O)C2)ccc(C)c(C)c1 c1(CC)cnc(O)c(C(N2CCCCC2CCN(C(=O)C(C)OC(C)C)C)=O)c1 n1(CCC(=O)OCC)ccc(=Nc2nnc(C(O)CC)n2CC(C)C)[nH]1 N1(CC)CC2CN(C(C3CN(C)CCN3C(c3cc(COC)on3)=O)=O)CC2C1 CC(C)(C(=O)N1CC(C(F)(F)F)C(CNC(c2ccno2)=O)C1)S(=O)(=O)C1CC1 C1(N(C)C(c2ccc(O)nn2)=O)CCCN(Cc2csc(-c3cccs3)n2)CC1 N#CC1CCN(C(C2CC23CCN(Cc2ccc(-c4cc[nH]n4)cc2)C3)=O)CC1 N1(C(C=C(C)C)=O)CCN(CCCCC2CCCN(C(=O)C(=O)N(C)C)C2)CC1 C1(C(C)NC(C2(F)CCC2)=O)CCN(C(=O)Cn2cnnc2O)C1 CCC(C(=O)NCC(C(=O)NCCC(C)C)OC)N(C)C C1(C)(C(N(C)Cc2ccc(C)s2)=O)CC12CCN(CC(=O)NC(C)(C)C)CC2 c1(CC(N2C(CNC(=O)CN3CCCCC3=O)C=CC2)=O)ccc([N+](=O)[O-])cc1 CC1=C(C(=O)NCCCCC2CN(C(C3(O)CCOC3)=O)C2)CCO1 C#Cc1cccc(C(=O)NCCC(C)N(C)C(C2CCC3C(C2)C3(F)F)=O)c1F c1(-c2nc(C(C)C)nn2-c2ccc(OC(F)(F)F)cc2)cn2ccccc2n1 C1(NC(C=CCNC(C(C)NC=O)=O)=O)CC12CCCC2 C(=O)(C1=Cc2cc(F)ccc2OC1)N1CCC(N(c2ccnc(C)n2)C)C1 N1(C(=O)OC(C)(C)C)CC(F)(F)CC1C(N1CCC1Cc1cn(C(N)=O)nn1)=O C1(c2noc(-c3ccc(OCC(C)C)o3)n2)(NC(C(CC)SC)=O)CCCCC1 N1(C(C(CC2CC2)NC(c2cc(Cl)cs2)=O)=O)CCCC2(C1)N=N2 N1(C(C(CC)COC)=O)CC2CCCCC2(CN=c2[nH]c(Cl)ncc2Cl)C1 CN1C(=O)CCC1C(=O)NCc1c[nH]nc1C1CCN(C(=O)CC2CC2)C1 N1(C(CCOCCOC)=O)CCC2CCCC12C(=O)NCCC1CC(=O)N(C)C1 C1(C(=O)NC2COC3(CCC3)OC2)Cc2ccccc2S1(=O)=O N1(C(C23N(C(C(C(CC)C)N(C)C)=O)CC(C2)C3)=O)CCOC2COCC12 C1(C(=O)NCCCCCN(C)CC)C2CC(O)C(C2)N1C(=O)C1=CCCC1C N1(CC(=O)N(CC(CNC(COCCOCC)=O)C)C)CCCNS1(=O)=O n1(CC)ccc(=NC(=O)C2=CCCN(C(=O)C(C(C)C)OCCOC)C2)[nH]1 c1(N2CCN(CC(C)O)CC2)nc2ccc(Cl)cc2c(=NCC2(C)CC2)[nH]1 CS(=O)(=O)c1ccc(C(N2CC(O)CC2C(=O)NCCc2ncc[nH]2)=O)cc1Br c1(CSCC)cn(C2CCC(C(=O)NC3CS(=O)(=O)C3)C2)nn1 Clc1cccc(CNCC2COC2c2ccccc2)n1 c12ccc(cc1)OCC2.C(=O)(CC(=O)OC)NCC(C)NC(COC)=O N1(C(c2nccn2CCC)C(=O)NCC(=C)C)CCOC(C)(CC)C1 CC(C)(C)CC(=O)NCC1(F)CCN(C(C2(CN3CCCC3)CCCC2)=O)C1 N1(C(CN(C(C)C)C)=O)CC2CCC(C1)C2NC(C1CCCC(=O)N1)=O C1(C2CC2)(CNC(C(F)=CC)=O)CCN(C(=O)C(c2ccccc2Cl)C)C1 c1(CC)cccc(C(N2CCN(C(=O)C(n3nc(C)cc3C)C)CC2)=O)c1N CC(C)(C)[Si](C)(C)OCc1ccccc1.C12(CCC1)C(=O)N(CCO)CCCO2 C1(NC(CC(=C)C)=O)CCC(CNC(C2(C)CCCO2)=O)CC1 c1(OCCCC)ccc(CCN(C2CCN(C(=O)C(C)CC)CC2)C)cc1 c1(C(=O)NC2CC(O)(CNC(C3(OCC)CCC3)=O)C2)cc(C)c(C)cn1 C1(OC)CN(C(c2cccc(C(C)C)n2)=O)CC1NC(=O)C(F)=C1CCC1 N1(C(C=NOC)=O)CCOCCC1C(=O)NC(C)COC(C)C C(C)(C)(CC(=O)NC(C)CCO)N(C(=O)Cc1ccon1)C N(C1CN(C(c2ncc[nH]c2=O)=O)Cc2ccccc21)C(C(CCC)N(C)C)=O N1(C(=O)CCCN2CCOCC2)CCC2(CCCN(C(=O)CCC3CC3)C2)C1 Cc1cnc(F)cc1C(=O)N(C)CC1CCCN1C(c1ncc(C(F)(F)F)s1)=O C12(CNC(CCc3c[nH]c(=N)[nH]3)=O)CCC1CN(C(c1ccc(Cl)cc1Cl)=O)C2 c1(-c2ccc(CC(=O)NC(=O)NCCCOC)cc2)ccc(C(F)F)c(F)c1 CCCCC(C)CCC(=O)OC1CCCCC1SCC1=NOC2OCCC12 C1(C)(OC)CCN(C(c2ccc(-c3cn(C)nc3C)cc2)=O)C1 C#CCC(C(=O)Nn1cnnc1C)NC(=O)CC(C)(C)C=C c1(OC)cncnc1C(=O)NC1(C(=O)NCC(C2CCCCC2)O)CCC1 C1(CC(=O)OC)CCN(C(=O)C(C2CCN(C(=O)CSC)C2)F)CC1 Cc1c[nH]nc1C(=O)NC(C)CC(=O)NCCCSCCO C1(CC(=O)NCCC2(NC(=O)CN(C3CCC3)C)CCC2)(OC)CCC1 C(=O)(C(C)(C)C#N)NCC1C(C(=O)NCc2cn(CCC)nn2)CC1 C(=O)(CC(C)C(F)F)NCC(CC)NC(=O)Cc1ccccc1C1CC1 C1(N(C(c2ccc(C(C)C)o2)=O)C)CN(C(c2coc(O)n2)=O)CC12CC2 C1(NC(CNC(=O)OC)=O)CCC2(CC1)CN(C(=O)C1=CS(=O)CCC1)CCO2 c1(C(N2CCN(C(C3CC(SC)C3)=O)C3(C2)CC3)=O)cc2c(C)cccn2n1 c1(C(C(=O)NCc2cccs2)N(CCCC#C)C)nocc1CC CC(C)C(C)C(=O)NCC1CC1NC(c1cc(Br)cn1C)=O C(=O)(C1=CC2C=CC(C1)C2)NCCCC1(NC(C(C)C(F)(F)F)=O)CCCCC1 N1(C(C(C)O)=O)CCC(C)(CCNC(=O)Cc2csc(NC=O)n2)C1 c1(OC(C(N2C(CNC(C3(OC)CCCCC3)=O)CC2)=O)C)ccc(Cl)cc1C c1(NC)snc(C)c1C(N1CC2CC2(NC(=O)CC2(CO)CC2)C1)=O N1(C(c2c(CC(=O)OC)occ2)=O)CC2(CCCC2NC(=O)CCCC(C)O)C1 Cc1ccc(CCCCC(=O)NCC2C=CCN2C(C2C3CNC(=O)C23)=O)cc1 C=C(C)CCC(=O)N(C1CCCCC1NC(=O)Cc1nc(C)sc1Cl)C C(=O)(CC(C)(C)C1CC1)NC(C)CCNC(C1CCCN1C1CCOCC1)=O C1(NC(Cc2n(C)cnc2)=O)(CNC(=O)CCF)CCCCCC1 C1(CNC(c2ccc(O)nc2)=O)CC2CCC1N2C(=O)CCC1CCC1 C1(C(CNC(=O)Cc2nc[nH]n2)F)CCN(C(=O)CCc2nncs2)CC1 C1(NC(C(F)=CCC)=O)CCN(C(c2cnnc3sccc23)=O)CCC1CO C(=O)(C1Cc2ccc(Cl)cc21)N1CC(F)CC(NC(CC(C)C)=O)C1 N1(C(c2c(CC)csc2)=O)CCN(C(c2ncn(C(C)C)n2)=O)C(C)C1C c1(C(=O)NC(C)(C)CCNC(C2CC2Cl)=O)cc2c(cc1N)OCO2 N1(C(COC(c2nccn2C)C)=O)CCC(NC(c2cncs2)=O)C(O)C1 C12(CNC(c3cnc(CC)s3)=O)CC1CN(C(=O)C(CC)C1CCOCC1)C2 c1(C(=O)NC(CNC(C(C)OCCCC)=O)C(C)C)cccc2nc(C)cnc12 C1(C(=O)NC(c2ccnn2C)C(=O)N(CC(O)COC)CC)CC2CC2C1 C1(c2onc(-c3nccc(N)c3)n2)CC2c3ccccc3C1c1ccccc12 CCCC(C(O)C(=O)N(C)CCc1ncon1)NC(C1CC(F)(F)C1)=O C1(NC(CN(C)C2CC2)=O)CCN(C(c2cc(=O)cc[nH]2)=O)CC1F c1(C(=O)NCCCN(C(=O)C(F)F)C2CC2)ccccc1C1CC1(F)F C1(C(=O)NCCC(C)(C)NC(=O)C(O)C2CC2)CCc2ccnn2C1 C(=O)(C1=NOC(C)C1C)NC1(C(=O)NCc2c(C)nn[nH]2)CCC(C)(C)C1 c1(C(C)C)ccc(CN2CCCC(c3cn[nH]c3)C2)cc1F C1(C)(C(=O)NC2CCCN(C(C)=O)C2)CN(C(=O)C(C)n2cnnn2)C(C)(C)C1 Cc1ccc(C(N2CCCOC(CCNC(=O)C(F)(F)C(C)O)C2)=O)c(F)c1 C(C)(C(CC(=O)NCCC(O)CO)NC(=O)CC1CC(C)=NO1)OC C(=O)(C1=NOC2COCC12)NCC1CCC(NC(c2[nH]cc(CC)c2)=O)CC1 c1(COC)ccc(CC(=O)NCCC2CCC(NC(C3(CF)CCC3)=O)C2)cc1 n1(CC)cc(C(=O)NC(C)(C)CN(C(=O)CCCCOC)C)c(C)n1 CC(C)C(CCNC(=O)CSCC(N)=O)NC(c1csc(-c2ccccc2)c1)=O c1(C(=O)NCC(C2CC2)NC(CC(=C=C)C)=O)sc2cccc(F)c2c1COC C1(C(=O)NC(CN(C(c2ccc(C)c(C)c2)=O)CC)C)CC2COCC2C1 N1(C(C2CNCC(C)(C)S2(=O)=O)=O)CCOc2cccc(F)c2C1 N1(C(C2(C)C(C)CCC2)=O)CCC2(CCN(C(=O)C(c3csc(=N)[nH]3)=O)C2)C1 N1(CCCC(=O)NC2CC(O)C2)C(=O)CCC1=O C(=O)(C1=C(F)CN(C(C2CCCCNC2=O)=O)CC1)NCC1(O)CCC(C)C1 c1(C(C)C)nc(NCc2cccnc2)cc(=NCC(CC2CC2)CO)[nH]1 C1(NC(C(c2ccc(-c3cnco3)cc2)N(C(C=C)C)C)=O)CCCCCC1 CC1(C(=O)NC2CCC(NC(=O)C(c3ccc(F)cc3)(C)F)CC2)COC(=O)C1 n1(COC)ccc(C(=O)NCCN(C(=O)Cc2ccsn2)C(C)C)n1 S(=O)(=O)(c1c[nH]ccc1=NC1CCN(C2CC2)C1)N1C(C)(C)C=CC1 N1(C(c2c(N)cc(OC)cc2F)=O)CCCC2(CCCN2C(C2CC23CC3)=O)C1 C(CN=c1[nH]c2c(c(=NCC3(C)CC3(C)C)[nH]1)SCC2)c1n(C)ncn1 c1(CC(=O)NCC2(O)CCN(C(C3C(CC(C)C)C3)=O)C2)c[nH]c2cccnc12 N=c1[nH]cncc1CN1CCOC(C(=O)NCC=CCl)C1 C1(C(=O)NCC(C)N(C)C(C2CC3CCC(C2)C3O)=O)CC(C)(C)OC(C)(C)C1 Cc1ccc(F)cc1C(=O)NC(CNC(c1cc(O)ccc1F)=O)C(C)(C)C c1(NC2CC(CNC(Cc3nc(C)sc3C)=O)C2)cc(C)c([N+](=O)[O-])cc1Br c1(C(=O)NCC(N=c2[nH]nco2)c2ccccc2)ccc2c(c1)CCCCN2 N1(C(CCC(CC)CC)=O)CCC2(CCCC2NC(=O)Cc2cncn2C)CC1 C(CC(C)(C)C(F)(F)F)NC(CS(=O)(=O)N(C)C)C1CCCC1 C1(NC(c2ccc(CC)cn2)=O)(CNC(=O)Cc2c[nH]nc2C)CCCCCC1 C(=O)(CC(C)C(F)F)N.C1(C(=O)NCCN(CC)CC)CC12CC(NC(C)=O)C2 N1(C(C(C)OC(C)(C)C)=O)CCC(C)(C(=O)NC2CN(C(N)=O)C2)C1 Cc1cnc(C(=O)NC(C)CCNC(C2CC2CC(F)F)=O)o1 C1(CNC(C2(C(=O)OCC)CC2)=O)CN(C(C2CCCC2)C)CCO1 C=CC(C)(CCOC)C(=O)N1CCN(C(=O)C(CN(C)C)CC)C(CCO)C1 N1(c2nnc(C(=O)OCC)s2)CCC(CNC(c2cnc[nH]2)=O)C(C)C1 N1(C(C(CC)O)=O)CC(OC)CC1CCNC(c1n[nH]cc1C)=O N1(C(C(c2ccc(N)cc2)C)=O)CCC(C(C)NC(C2CCSC2)=O)CC1 C1(OC)(CNC(C2CCC2)=O)CCN(C(=O)C(C)(O)C2CC2)C1 C1(CNC(CSCC(C)=O)=O)C2CN(C(C3(C)CC3c3ccccc3)=O)CC12 c1(NC(c2cn(CCNC(C3CCCS3)=O)cn2)=O)ccc(O)c(Cl)c1 C1(C(=O)NCC(O)CCNC(c2cnc(Cl)n2C)=O)(OC)CCCOC1 c1(OC)cc(-c2ccsc2C(=O)Nc2cc(C)cnc2Br)c([N+](=O)[O-])cc1OC C1(C(=O)OC)C2CCC1(c1nccs1)C2.C1(=O)C(NC(C)=O)CSC2CN1C2 C(=O)(C(C1=NOC2CC12)N1CCc2nc(Br)sc2C1)NCCCCCC CCC(C)(CO)C(=O)N1CCC(C)(CNC(C2(c3cccc(OC)n3)CC2)=O)C1 n1(C(C)(C)C)nnnc1C1C2(CC2)CN1.C1(C(C2CCCC2)OC)CCCCC1 O=C(C1=CCCOCC1)NC1CC(O)CN(C(C2(C(F)(F)F)CCCCO2)=O)C1 c1(C(=O)NCC(CC(=O)OC)C)n[nH]c2c1CN(C(C1(CC(C)C)CC1)=O)C2 c1(N(CC(C2CC2)OC)C)nc(=NCCC(C)(C)C)[nH]c2c1COC2 c1(CNC(c2cncc(-c3cc(F)ccc3Cl)n2)=O)ccc(C(=O)O)cc1F C(CCCC(=O)N(C)C)c1nc(CC(C)N=[N+]=[N-])on1 CCCC(C#N)C(=O)N1CCC(NC(C2CN(CC)CCO2)=O)C1(C)C C1(NC(C(C)NC(N)=O)=O)CCCN(Cc2ccc(C(C)C)s2)CC1 C(=O)(C#CC1CCOCC1)NC12CC(NC(C(C)(Cl)Cl)=O)(C1)C2 N#CC1CCN(C(c2cncc(NC(=O)Cc3cc(Br)cs3)c2)=O)C1 CC1CCCN(C(C2CCCN(C(C3CCOC3)=O)C2)=O)C1CO Cc1oc(C(C)C)cc1C(=O)NC1CC(C)(NC(=O)CCCn2cccn2)C1 Cc1cc(F)c(C(N2CC(NC(c3cc(O)nc(Cl)c3)=O)C(F)C2)=O)cc1F c1(C(=O)NC2CCN(C(c3n(CC(C)C)ncc3)=O)C2)ccc2nccn2n1 C1(CC)CN(C(=O)CS(=O)(=O)NC)CCC1NC(C1CCCCC1O)=O N1(C(C(C)OC(C(C)CC2CCCO2)=O)=O)CCc2ccccc2C1 CC12CC(C1)C(C(N1CCC(NC(=O)COc3ccc(F)nc3)CC1)=O)CO2 c1(C(=O)NCC2CN(C(c3cnc(C)nc3)=O)C2)c(Cl)cccc1I C1(F)(C(=O)NCC2(OC)CC2)CCCN(C(=O)Cc2c(C)cnn2C)C1 Cc1c(C(N2CCC3CC3(NC(=O)C3CC3)CC2)=O)sc2cc(F)ccc12 CCCCC(C(=O)N(C)CC1CCN(C(=O)C(C)(C)C2CCOC2)CC1)N(C)C n1(CC(=O)NCC2(F)CN(C(C3=C(C)OCCC3)=O)C2)ccc2ccc(Cl)cc12 c1(N(C)C)cc(Cl)cc(Cl)c1C(=O)NC1CN(C(C2(C#N)CC2)=O)CC1C#N c1(C(=O)NC(C)CNC(c2ccn(C)c2)=O)cc2cc(F)c(F)cc2[nH]1 CC1CC2CN1C(=O)C1(CC1)C(=O)NC2.c1(C(=O)OC(C)(C)C)ccc[n+]([O-])c1 C1(NC(c2cnc(C)n2C)=O)C(C)CN(C(C2(c3ccncc3)CC2)=O)CC1C C=CC1CN(C(c2c(C)nn(CCC)c2C)=O)CC1NC(=O)CCCNC(C)=O c1(CN(C)C(c2ccnc(C3CCCC3)n2)=O)cccc(Cl)c1Cl n1(CC#C)cc(NC(C2CC(C)(NC(=O)C(O)COC)C2)=O)cn1 C1(C(N(CCCCCCNC(C(CCC)C)=O)C)=O)CC2CCCCC12 C1(NC(N2CCN(Cc3ccnc(OC(C)C)n3)CC2)=O)CCCC2(CCC2)O1 c1(C(=O)NCC2C(C)(C)CN(C(=O)CC34CCCC3C4)C2)ccsc1S(C)(=O)=O C(N=c1[nH]c(=NCCS(C)=O)[nH]c2c1CSC2)C1C(C(C)C)C1 c1(C(=O)NC2CN(C(CCOCC)=O)CC2N=[N+]=[N-])c[nH]c2cccnc12 c1(OC)ccc(C)nc1C(=O)NC(C)(C)CNC(=O)C(C)Cc1cccc(Cl)c1 CC1(CNC(C2CC3C=CC2O3)=O)CN(C(=O)CCCc2ccsc2)CCO1 CCC(C(=O)NC(C)CNC(c1cc(-c2ccccc2F)[nH]n1)=O)C(C)(C)CC CC1(CCCO)CCCN1C(C1CC=CCC1NC(C1CC2(CC2)C1)=O)=O c1(C(=O)NC(CC)COC(F)(F)F)coc2cccc(O)c12 c1(CN(C(=O)NC2CCN(C)C2)CC)cc(OC)c(Br)c(OC)c1 c1(C(N2CC(C(=O)NCCN)OCC2)=O)ccccc1[N+](=O)[O-] C1(C(=O)NC(CNC(C(n2ccc(C3CC3)n2)C)=O)(C)C)C2COCC12 c1(CC)ncc(NC(=O)CCN(C(C2SCC=C2C)=O)C2CC2)cn1 C(CNC(c1cn(C)nn1)=O)(CC(F)(F)F)NC(CCN(CC)CC)=O C1(C(=O)NCC(C)(CO)NC(C(C)C#N)=O)CN2CCN1CC2C CC(C)(C(=O)NCCCN(C(C1COC(=O)C1)=O)C1CC1)c1cnc[nH]1 N12CC3CC3(C1)C2.C1(S(N)(=O)=O)(CCc2cn(CCC3N(C)CCC3)nn2)CC1 C=CC(C)(O)C(=O)NCC1CC(C)N(C(=O)C=Cc2cn(C)nn2)C1 N1(CC)CCN(CCC(N2CCC(NC(=O)CC3CCCC(=O)O3)C2)=O)CC1 C(=O)(C(C)(C)NC(=O)C(F)(F)F)NCC(CC)NC(=O)C(CO)NC(=O)C1CC1 Cc1ncc2ccc(C(N3CCC(O)C(NC(C4CC=CCC4)=O)C3)=O)cn12 Cc1nnc(NC(C2CN(C(c3ccnc(Cl)c3)=O)CCO2)C)c(C#N)c1C N1(C(c2n(COC)ncc2)=O)CC(CCNC(C2(CO)CCCC2)=O)OC(C)C1 c1(OCCCCC)cc(NCc2cncc(CC)c2)ccc1C CC1Cc2c(C(=O)O)cccc2CN1C(=O)CCn1cc(C(N)=O)nn1 c1(C(=O)NC(CNC(c2n(CC)nnc2)=O)CO)cc(S(C)(=O)=O)cc(C)c1C n1(CC(=O)NCC2(CNC(CC=CCC)=O)CC2)cnccc1=O N1(C(C)C)CC(N(C2CCC2)C(C2CC(O)(CN(C)C)C2)=O)CC1=O C(c1cccn1C)=CC(=O)NCC1CCC(NC(C(n2cc(C)nc2)(C)C)=O)C1 C(C1=CCN(C(c2ccn(C)c2CC)=O)CC1)NC(C(CC)F)=O c1(C(N2CCC23CCC(C(N)=O)CC3)C(=O)NC)ccc2cc(Cl)ccc2n1 CC1(C#CC(=O)NCCC2CCN(C(c3scc(Br)c3Cl)=O)C2)COC1 c1(C(=O)NC2CCN(C(c3cnnc(Cl)c3)=O)C2)cc(O)nc(O)n1 c1(CN2CCN(C(COC(c3c(C)nc(C)s3)=O)=O)CC2)ccc(O)c(F)c1F S(=O)(=O)(c1cc2cc(Br)cnc2o1)N1C(C)CCC(C(=O)OCC)C1 C1(C(=O)NCCNC(c2cc(CC)c(O)cc2)=O)Cc2ccccc2C1C C1(C(N(C(CCNC(Cc2nc(C)sc2C)=O)C)C)=O)CCC(C)(O)CC1 C1(NC(C(c2ccc(F)cc2)C)=O)CC(O)CN(C(=O)CCc2cccs2)C1 C12(C(=O)NCC3(O)CN(C(Cc4nnn(C(C)(C)C)n4)=O)C3)CCC(CC1F)C2 c1(C(=O)NC2(CCNC(C=CC)=O)CCCC2)ccc2nccnc2n1 C(=O)(C(CNC(C1(C2(O)CCC2)CC1)=O)C(C)C)NC(C(=O)OC)CC1CC1 N1(c2nc(=NCc3cn(CC)nn3)[nH]c(C)c2)CCOC2(CCOCC2)C1 Cc1ccc(Br)cc1CNC12CC(C(=O)NC3CCC(CO)CC3)(C1)C2 C(=O)(C(C)(C)CC(F)F)NCC12N(C(Cc3cccc(C)c3)=O)CCC1CC2 Cc1ncc(C(N2CC(F)(C(=O)NCc3ccc(C)c(C)c3)C2)=O)c(C)n1 c1(CN(CCNC(c2c(CC)scn2)=O)CCOCCO)cccc2cncn12 Cc1nc2ccccn2c1C(N1CCC2(NC(C3CCC=CCC3)=O)CC2C1)=O CN=c1[nH]c(=NCCN2CCC3CC23)[nH]c(=NCCCCC(F)(F)F)[nH]1 N#Cc1cncc(CC(=O)NCC2CN(C(=O)C3CC3)CC2(F)CO)c1 C1(C(=O)NCCCN(C(C(N2CC(C)C2)C)=O)CCO)(C(F)F)CC2(CC2)C1 c1(C(=O)NCCC(C)NC(C=Cc2c(C)coc2C)=O)cccc2nccn12 CCCCC(F)C(=O)N1CC2CC(C(=O)NCCc3[nH]cnc3C)(C2)C1 Cc1[nH]c(=N)sc1C(N1CCC(CN(C)C(C2CCCC2)=O)C1)=O N1(C(CCCC(CC)NC(c2c(C)nsc2C)=O)=O)CCC2CCN(C)CC12 c1(CCC(=O)NC(CC=C)CNC(C2CC(OC)C2)=O)ccc(Cl)c(OC)c1 c1(C(C)=O)cc(C(N2CCN(C(=O)CC3CC(C)=NO3)C(CO)C2)=O)ccc1O c1(C(=O)NC2(CO)CN(Cc3ccc(C)cc3F)C2)cc(F)c(F)cc1O C(=O)(C(C)CCCCCC)N1CCCCC(C(N(CCCC#C)C)=O)C1 CC1CN(C(=O)NC(C2C3COCC23)C(=O)O)CC(C)C1C(=O)OC(C)(C)C c1(C(=O)NCC(F)CNC(c2ccc(CO)s2)=O)cc(F)c2cn[nH]c2c1 c1(OCCC)ccc(N(C)C(c2[nH]cc(C(C)=O)c2C)=O)cc1 C12(CC(=O)N(CCC(C)NC(c3cnc(SC)s3)=O)C)CCC(C)(C1)OC2 N1(C(c2cc(C)c(C#N)cc2)C(=O)NC2CCC2)CCn2nc3c(c2C1)CCC3 N1(C(C(C(C)C)n2cncn2)=O)CCOC2(CCCN(CCc3cnco3)C2)C1 c1(SC2N(C(c3c(C)scc3)C(=O)NC3(C)CC3)CCCC2)cccc(Cl)c1Cl C1(NC(C2(CC=C)CCCC2)c2nnnn2Cc2cccs2)CCC(=O)N(C)C1 CC(O)(CNC(C1(NC(=O)COCCCN=[N+]=[N-])CCSC1)=O)CCO C1(NC(C(CSC)O)=O)CC(C)CN(C(c2cc(C)n(C(C)C)c2C)=O)C1 N1(C(CCC(C)SC)=O)CC(CNC(c2ccncc2F)=O)OC(C)(C)C1 O=C(CCCS(=O)(=O)c1ccc(Br)cc1)Nc1cc(OCC(F)(F)F)cc(F)c1 CCCCC(C)N(C)C(c1ccc(CNC(C2SCCS2)=O)s1)=O C1(N(C(Cc2nc(C)sc2)=O)C)CCCC(NC(C2(CO)CCOCC2)=O)C1 c1(C(N(CCCN(C)C)CCNC(C(C)C)=O)=O)ccc2ccnn2c1 c1(NC(c2cccc(OC)n2)C)nccc(=NC(C)c2ccc3c(c2)CCN3)[nH]1 c1(C(C(=O)NCC(CC)(C)NC(=O)CN2CCC(C)(C)C2)C)cc(C)cc(F)c1 N1(C(=O)Cc2cscn2)CCCC1CCc1cn(CCN2CCCCC2)nn1 C1(C(N(C2CCN(C(=O)COC3(C)CCC3)C2)C)=O)CCc2nnc(O)n2C1 c1(CC(C)C)ccc(C(=O)N(CCNC(=O)C2=CCC2)C(C)C)s1 C1(C(=O)NC2CCCCCC2)CCCN1NC(=O)C1CC=CCC1 N1(C(c2c(C)nn(C)c2)=O)CCCC(C(=O)NCC(C)(O)C(C)C)CC1 C1(CC)CN(C(=O)Cc2n[nH]c(C)n2)CCC1NC(=O)C=CCCC=C(C)C c1(N(C)C)cncc(C(N2CCCC2(C)CNC(=O)C(F)F)=O)c1 C1(C(=O)NC(C)C(=O)N(C)C)C=CCCN1C(=O)Cc1ccco1 c1(CC(=O)NCC2C(NC(C3(CC(C)C)CC3)=O)CC2)nc(C(C)(C)C)cs1 N1(C(CCNCC)=O)CC2C3CCC(C3)C2C1.C1(C=O)CC=CC(O)C1 CC1COCC(C(=O)NCc2cnn(C)c2C(=O)NCc2ncc(Cl)cn2)O1 N1(C(C(CC)NC(C)=O)=O)CCC(NC(=O)Cn2cncn2)CC12CCCC2 c1(NC(C2CCN(Cc3ccc(COC)s3)C2)=O)ccc(OC)c(OCCO)c1 CC1CCCCC1C(=O)NCCCOCCC(=O)NCCC1CC1 C(=O)(C(CCF)NC(C1CCCN1c1ccccc1)=O)OC C1(CNC(C(=O)NCC)=O)CN(C(=O)C(CC)C2CCOCC2)CC1(C)C C1(C(=O)NCC(CC)N(C)C(c2nnsc2C)=O)C2CC3C(C2)C13 c1(OC)cc(NCC2(O)CCC(C)(C)CC2)c([N+](=O)[O-])cc1F c1(CC(=O)NCCCN(C)C(C2(C#N)CC2(C)C)=O)ccc(Cl)c(F)c1 CC1CN(C(=O)CN2CC3CCC2C3)CC2(CCN(C(=O)C(C)CO)C2)O1 C1(CNC(C2C(F)(C(=O)OC)C2)=O)COCCN1C(C1CCC(OC)CC1)=O CC(C)C(C)CC(=O)N1CCC(C)(C)C1CNC(C1CCCCCC1)=O O=S(=O)(c1ccc(=NCCN2CC3CC3C2)[nH]c1)N1CCC2(CC1)CC2CO Cc1cc(N)ccc1C(=O)N(C(C)CNC(c1cccc(OC(C)C)c1F)=O)C c1(C(=O)NCC2N(C(C(CC)(C)O)=O)CCC2)ccc2[nH]c(=N)[nH]c2c1 CC(C(=O)N1CC(NC(=O)COCC(F)F)C1)c1cc[nH]n1 c1(NC(C2CCC(NC(c3cc(CC)nn3C)=O)CO2)=O)cc(O)c(Cl)cc1Cl c1(NC)ccc(C(=O)NCC(C)(O)CNC(=O)CSc2cccs2)cc1F CC1CCC(CCNC(C23CC(NC(=O)CSC4CC4)(C2)C3)=O)O1 N1(C(C(C)OCCOCC)=O)CCC(C(=O)NC2CCCC2F)C(O)C1 C1(NC(C=CCN(C)CC)=O)CCCC(NC(C2CCOC(C(F)(F)F)C2)=O)C1 Cc1c(CN2CCC(CNC(C3CNC(=O)O3)=O)C2)cnn1C c1(NC(=O)CCCCCCBr)cnc2c(c1)CN(C(=O)CCc1cnc[nH]1)CC2 n1(CC2CN(C(CSC)C)C2)nc(C(=O)NC2Cc3ccccc3C2)ccc1=O c1(C(N(C2CCN(C(C3CCC4CC3C4(C)C)=O)C2)C)=O)cc2n(c1)CCOC2 N1(C(c2c(C)cc(C)s2)=O)CCC(C)(C)C(NC(=O)Cc2cn(C)nc2C)C1 Cc1cnc(C)c(C(=O)NC2CCOCC2NC(=O)CC2CCC(=O)N2)c1 N1(C(c2c(C)nc(N(C)C)s2)=O)CC(NC(c2cn(C)c(=O)n2C)=O)CC(C)C1 C1(C(=O)NCCN(CCCC)C)CC(NC(=O)Cc2cccs2)C1(C)C N1(C(CC=O)=O)CC2CC2(C(N2CC(SC(F)F)C2)=O)C1.N(CC)CC S(=O)(=O)(c1ccc(OC(F)F)cc1)NC1(CC(=O)NC2CCC(C)C2)CCC1 C1(CC(=O)N(CCNC(=O)CC(C)C(C)C)CC)SC2=NCCN2C1=O N1(C(C(C(CC)O)C)=O)CCn2ncc(CNC(C3CS(=O)(=O)CCO3)=O)c2C1 C(=O)(C(C)C(CC)CC)NC(CC#C)(C)C(=O)N1CC2(C1)CN(CC)C2 C1(CNC(CSCC(C)C)=O)CCCCCN1C(=O)CCN1CCCC1 C=CCC(CC=C)C(=O)N1CC(C(=O)NC2CCCC2F)C(C=CC)C1 n1(CCC=C)nc(-c2cccc(OC)n2)nc1C1C(C)CC1C N1(C(Cc2c(C)occ2)=O)CCCC(CNC(=O)CC(C)(C)C2CCCCC2)C1 CC1(C(=O)O)CCCC1NC(C1CC1C(N)=O)=O Cc1cccc(SCC(=O)NC2C(NC(c3cnn(C)c3)=O)CCC2)c1C Cc1cc(O)c(F)cc1NC(C1(C(C)C)CCN(C(c2cc(C#N)c[nH]2)=O)C1)=O N1(C(C)=O)CC(O)(C(=O)NCCOCCC(C)C)C1.C1CCCO1 C(=O)(C1=CCC(C)(C)CC1)N(CC(C)O)CCNC(c1cnc2ccsc2c1)=O C1(NCc2c(C(=O)OCC)ccs2)CCCC(NC(c2cnc(Cl)s2)=O)C1 C(=O)(CC(F)(F)C(F)F)N(CC(C)N(C(Cc1c(OC)ccc(Cl)c1)=O)C)C Cc1csc2c(N3CCC(O)(C(=O)NCCSC(C)(C)C)CC3)ncnc12 C1(C)(C(c2nnnn2C(C)C)NC(c2n(CC)ncc2)C)CCCCCC1 C1(C2CC2)(C(=O)NC(CCCC)CC)CN(C(c2cncs2)=O)C1 c1(C(C)C)ccccc1C(C1CC=CC1)N(C)C.C12CC(C1)C(=O)N2 C(C(C)(C)C(=O)N1CCCC(NC(c2c(C3CCC3)cnn2C)=O)C1)OC c1(C(=O)NCC2N(C(CN(C(COC)=O)C)=O)CCC2)cc(Cl)cc([N+](=O)[O-])c1 c1(CCC)ccc(C(=O)NC(CNC(c2nnn(C)c2N)=O)CC)cc1[N+](=O)[O-] Cc1cccc2cc(C(N3CCC(F)(CNC(C4CCCC4O)=O)C3)=O)nnc12 C1(C(=O)NC(C2CN(C(=O)C(F)(F)C(C)O)C2)C)Cc2cccnc2C1 Cc1nc(Cc2ccccn2)sc1C(=O)N(C1CN(C(=O)C(C)C#N)C1)C c1(C(N2CCCC(CNC(C(CCC)F)=O)(CO)C2)=O)cc(C)c(F)c(C)c1 N1(C(c2n(C)c(S)nn2)=O)CC(NC(=O)Cc2cc(F)ccc2O)CC(C)(C)C1 C1(CN(C(c2scc(OC)c2)=O)C)CCCCN1C(C1COCC1(C)C)=O C1(NC(C(C)N(C(=O)CCC2OCCO2)C)=O)CC(=O)N(C2CC2)C1 C=CCC(CC(C)C)C(=O)N1CCC(CCC(=O)Nc2cnc3[nH]cnc3c2)C1 C1(CNC(C2(OC)CCOC2)=O)CC(C(=O)NCCN2CCCC2)=NO1 CS(=O)(=O)c1cc(C(=O)NC2CC(NC(C3C=CC=CC=C3)=O)C23CCC3)cs1 c1(SC)cccc(NCCCCNC(=O)C=Cc2ncc(C)[nH]2)c1[N+](=O)[O-] c1(NC(C(c2ccc(C#N)cc2)O)=O)cccc2ccc(Cl)nc12 c1(NC(C2CC2C(N2C(COC)COCC2)=O)=O)cnc(Br)c(I)c1 N1(C(CCc2ncc(C)[nH]2)=O)CC2CC(C1)C2N=c1cc(Cl)nc(C2CCC2)[nH]1 c1(CC(=O)NC(CCN(CC)CC)C)ccc([N+](=O)[O-])c(N)c1 O=C(C=Cc1cncs1)NN1CCCC1C(=O)NC1(C2CCCCC2O)CC1 c1(CNC(c2cn(CC=C)nn2)=O)ccc(CNC(C2(C(N)=O)CC2)=O)cc1 CCC(C)CC(C(=O)NCC1CCC(=O)NC1)NC(=O)CCC(C)(C)N(C)C C=C(CNC(=O)Cc1cnn(-c2ccccc2)c1)CCNC(C1CCC(F)C1)=O C1(CCC#C)CCCN1C(C1OCCC1OC(C)=O)=O C1(OC)C(NC(c2cccnc2CNC(=O)C(=O)NC2CC2)=O)CC12CCC2 CC(C)CC(C)CNC(C1CSCN1C(C1CCN1C)=O)=O N1(C(c2c(C)scc2)=O)CC2CCC1C(NC(C1CC(C)C1C)=O)C2 c1(C(=O)NCC(CNC(c2cnn(CC3CCCC3)c2)=O)F)cncnc1 c1(C(=O)NC2(C(N(C)CC3C(C)C3)=O)CC(F)(F)C2)cncc2[nH]ccc12 c1(C(=O)NCCN(C(=O)CC(C)(F)F)C)[nH]c2ccccc2c1C1CC1 C1(NC(C2CCSCC2)=O)CCC2CN(C(=O)Cc3cnn4c3CCCC4)CC2C1 c1(C(N2CC(NC(C=Cc3cnc(C)s3)=O)C(O)C2)=O)ccc([N+](=O)[O-])cn1 c1(N2CC(C)C(NC(=O)C(F)F)CC2)nc2cc(F)ccc2o1 c1(C(N2CC(NC(COCC)=O)CC3(C2)CC3)=O)ccc2c(c1)CCN(C)C2 C1(C(N2CC(=CC)C2)=O)CC(OC)CN1C(C1CCCCS1)=O c1(OCCOC)cc(C(=O)NCC(F)CNC(=O)C(c2cncnc2)C)ccn1 C1(C(=O)NCC(O)C2CC2)CCCN(Cc2nc(-c3ccncc3)cs2)CC1 C1(C(=O)NCC2C(C)CN(C(=O)Cn3ncnn3)CC2)CC(=O)CC12CCC2 CCC(C)(COC)CNC(=O)CCC(C)NC(C1CC1(Cl)Cl)=O c1(C(N2CCC(CC=C)(NC(c3coc(CO)c3)=O)C2)=O)nc(=O)cc(N)[nH]1 N1(C(C2N(C(CC3ON=C(CC)C3)=O)CCCCC2)=O)CC2NC(=O)OC2C1 C(CCC1CC1)(C(=O)NC1CC1)NC(C(C)OCCCC)=O CCC(F)C(=O)N1CC(O)(C(C)NC(c2occc2CNc2ccccc2)=O)C1 c1(C(=O)NC2CCCCN(C(C(P(C)(C)=O)O)=O)C2)ccc(F)c2cccnc12 c1(OC)cccc2c1OC(C(=O)NC1CN(C(c3cc(F)ccc3O)=O)C1)C2 N1(C(C2C(CCC)CCC2)=O)CC2CC2C1C(=O)NCCCN(C)OC N1(C(CCCOCC)=O)CC(NC(C2CNC(=O)N2)=O)C(C)(C)C1 C#CCC(CC(=O)NCc1nc(C(N)=O)co1)NC(=O)C(C)(O)C(C)C C1(NC(C2(c3ccccc3)C(C)(C)C2)=O)(CO)CCN(C(=O)Cc2cc[nH]n2)C1 N1(C(C2CC(O)(CC#C)C2)=O)CCC(NC(=O)CC2CCCN2CC)C12CCC2 C1(C(=O)NCCCCC2CCCN(C(C(C)C#N)=O)C2)CCC(=C(F)F)CC1 c1(C(=O)NCCSCC(N2CC(CCO)C2)=O)ccc2c(c1)CC2 c1(NCc2cnc(C(C)(F)F)s2)nc(Cl)[nH]c2ncnc1-2 N1(C(c2c(C)nc(C)s2)=O)CCOCC(C(=O)NCC(C)(C)C2(O)CCC2)C1 C(C1OCCc2sc(C(=O)O)cc21)NC(c1c(OC)cc2c(c1)OCO2)=O CCCCCCN(CCCO)N1CCC(c2nc(Cc3ccccc3)cs2)CC1 c1(C(=O)NC2CCCC(C(=O)NCC3CC(F)C3)C2)cccc2c1CCCC2 CC1CN(C(c2cncc(N(C)C)c2)=O)CCN(C(=O)COCCF)C1 C1(C(N(C2CC(C)C2)C)=O)(NC(=O)CN=[N+]=[N-])CCCCC1 c1(C(=O)NC(C)CNC(=O)CCCc2ccc(Cl)cc2)cc(C(F)F)ccc1Cl C1(NC(C=C2CCC(C)CC2)=O)CN(C(=O)C(C)(C)N2CCCCC2)CCC1O N1(C(C(CC)Sc2nc(=N)[nH][nH]2)=O)CCCC(NC(=O)CCc2nc(C)cs2)C1 c1(C(=O)NCC(CNC(Cc2ccn(C)n2)=O)(C)O)ccc(N)c(F)n1 N1(C(c2c(SC)cccc2)=O)CC2CC(NC(c3cc(C(N)=O)co3)=O)C(C2)C1 C1(O)(CN(C)C)CCN(C(=O)NCc2cccc(N3CCCC3)n2)C1 CC(C)(O)C(F)C(=O)NCC1CCN(C(=O)CCCCc2ccc(Cl)cc2)C1 C1(CC)CN(C(c2sc(Br)nc2C)=O)CCN1Cc1ccc(OC(C)C)nc1 N1(CC(=O)NCC23CC2CN(C(C2CC4(CC4)C2)=O)C3)CCn2ccnc2C1 c1(C(N2CC(O)(C(C)NC(C(CSC)O)=O)C2)=O)noc2ncccc12 CON1CCC(CC(=O)NC2(C)CCCN(C(=O)CN3CCC(C)CC3)C2)CC1 C(=O)(C(C)(C)CCC#N)NCC#CC(=O)N1C(CC(C)C)CC1 C1(CNC(C2CCCC(C)O2)=O)CC2(CC2)CN1C(=O)CN1CCCCCC1 C1(C(C)C)CCC(C)CC1C(=O)NCC1(C(C)NC(C2(F)CC=CC2)=O)CC1 C1(C(N(C)CCO)=O)CN(C(=O)C=Cc2ccccc2Br)CC12CC2 C1(C(N(CC(C)(C)N(C)C)C)=O)CC2CN(C(C3(F)C(C)(C)C3(C)C)=O)CC2C1 C123CCC(C1)C(S(=O)(=O)C2)N(C1CCCS(=O)(=O)C1)C3=O C1(NC(CCC#C)=O)CCCN(C(c2nnc(S)n2C)=O)CCC1 Cc1ccc(Cl)c(C(=O)NC(C)CCNC(=O)CCc2ccoc2)c1 C1(C2CCC2)(C(=O)NCC2CC(F)(CN)C2)CCC1 C(=O)(CCCCCCC(C)=O)N1CCC(C)(NC(CC=C)=O)C1 CCCC(CCC)C(=O)N1CCN(C(=O)CCCCNC(C)=O)C(CF)C1 N1(c2nccc(OC)n2)CC2C(C1C(=O)Nc1ccc(C(N)=O)nc1)C2(C)C N1(C(c2ccc(CC)[nH]2)=O)CCN(C)CC1CNC(=O)C(c1c(C)noc1C)C C1(CC(=O)NCC#CCNC(C2C(CC)C2)=O)(CO)CCCC1 CC1(C)COCCC1CNC(C1CSCCN1C(=O)CCN1CCCC1=O)=O c1(C(=O)NCC2(COC)CCCN2C(c2cccnc2)=O)cn(C)c(=O)nc1O C1(F)(CNC(CC(C)CC(F)(F)F)=O)CC(N=c2nc(CC3CC3)[nH]s2)C1 C(=O)(CC1=CCCCC1)N1C2C(C(=O)OC)C(C2)C1.c12c[nH]nc1CNC2=O C1(F)(C(N2CCC(CNC(C(C)c3ccco3)=O)CC2)=O)C(F)(F)C1(F)F CC1CC(CNC(C2(C)CCC2)=O)CN1C(c1cc(C2CCOCC2)[nH]n1)=O C(=O)(C(C)(C1CC1)NC(=O)CCN(C)CCO)N1CC(OC)C1 Cc1c(CCC(=O)NC2CC2NC(C2CCCCNC2=O)=O)cccc1Br c1(C(N(C2CCN(c3nnc(CC(C)C)s3)C2)CCC)=O)coc(C(F)F)c1 c1(C(=O)OC)cc(CNC(C2(CNC(=O)CCc3ccsc3)CCC2)=O)cs1 CC(CCCCc1ccccc1)NCCCCF N1(C(CCCc2onc(C(C)C)n2)=O)CCCCC(NC(C2CCOC2=O)=O)C1 C(C(CC(=O)NC1(C)CN(C(C2(C)CCCS2(=O)=O)=O)C1)C(F)(F)F)N(C)C C=CC1CN(C(=O)C(C)(C)CNC(=O)CN(C)C(C)=O)CC1O CC(C(CO)NC(=O)CCCSC(C)(C)C)NC(=O)C(O)c1ccsc1 C1(CC(=O)NCC(CC)NC(=O)CCC2CCCCC2)COc2ccccc2O1 c1(C(N(CC(C)NC(Cc2c(C)noc2C)=O)C)=O)cnn2cnnc2c1 Cc1ccncc1CC(=O)NC1CC(CO)N(C(=O)C2=CCCS2)C1 n1(CCOC)cc(C(=O)NC2CCCCC2NC(=O)C(C)SC)c2ccccc12 c1(C(=O)NCCNC(c2c(NC)scn2)=O)cc(COC)oc1C N#CC1CCN(C(=O)C(C2CC=CCC2)NC(C2CCC3(CC3)C2)=O)CC1 O=C1CCC(NCC(N2CCC(CCC(=O)O)(C(F)(F)F)C2)=O)CN1 c1(C(N(CCN(C(c2c(C)nc(CO)o2)=O)C)C)=O)cc(S(C)(=O)=O)cnc1O CCC(C)(CCC(C)C)C(=O)N1CCC(F)C(NC(=O)CCN2CCCC2)C1 Cn1c(CN2CCOCC2CCS(C)(=O)=O)nc2ccccc12 CC1=C(C(=O)N2CC(C)(NC(c3cn4c(n3)CCC4)=O)C2)CCCO1 C1(NC(c2cccc[n+]2[O-])=O)CN(C(c2cc(F)cc(Cl)c2)=O)C2(CCOC2)C1 N1(C(CC)=O)CCCCC1CNC(c1cccc(OC)c1)=O N1(C(C(=O)Nc2ccc(NCc3cccc(F)c3)cc2)=O)CCOC2(CSC2)C1 c1(C(=O)NCCC2CCC(NC(CC(=O)NCC#C)=O)C2)csc2ccccc12 c1(C(=O)NCc2scc(C(=O)NCCCCCC=C)c2)ccnc(O)c1F C1(CCCC)CN(C(=O)C(O)C2CCCC2)CCN1C(=O)CCCC#N c1(CN(CC(c2nonc2N)=O)C)cn(CCC(=O)NCc2ccccc2)nn1 N1(C(c2cn3c(n2)CCC3)=O)CCCC12CCN(C(C1(C(F)(F)F)CCC1)=O)C2 Cn1cc(Br)c2c(NCC(O)C(F)(F)F)ncnc12 c1(SCC)cncc(C(N2CCC(NC(C3(CC(C)C)CCC3)=O)C2)=O)n1 c1(C(N2C(CNC(c3ccn(C)c3)=O)CCCC2)=O)ccc(C(C)(C)C)cc1N N#Cc1cnn(CC(N2CC3(NC(c4ccc(-c5cc[nH]n5)s4)=O)CC2C3)=O)c1 N1(C(CCCc2onc(C)n2)=O)CCN(C2CN(C(C3CC(O)C3)=O)C2)CC1 N1(C(c2c(CC)ncs2)=O)CC(C)(C)OCC1CNC(=O)C(F)OC(F)(F)F N1(C(CC(C)C(F)F)=O)CC2(CC(C(=O)NCCN(CC(F)F)C)CO2)C1 C1(OCC(N2CCN(CCNC(C3(C(N)=O)CC3)=O)CC2)=O)C#CCCCCC1 CC(C)C(C)(O)C(=O)NCc1cccc(NC(C2CCN2S(C)(=O)=O)=O)c1 c1(N2CCN(C(C(C)Oc3ccc(C(=O)OC)cc3)=O)CC2)cncc2nnnn12 Cc1ccc2[nH]c(C(=O)N(CC(C)NC(=O)CCc3cn(C)nn3)C)c(C)c2c1 C1(NC(C(CCOC)NC(c2ncccc2F)=O)=O)CCN(C)CC1C CN1CCCC(CCC(=O)N(C)CCNC(=O)C(F)=C2CCC2)C1 C1(CN(C(c2nc(COC)oc2)=O)C)C2CN(C(=O)C(F)=C(C)C)CC12 C(=O)(CC(C)C(F)F)NC(CCOCC)C(=O)NC(C)Cc1nncn1C N1(C(C(C)c2ccsc2)=O)CC(CN(C)C(c2cc(C(N)=O)[nH]n2)=O)C2(CC2)C1 C(=O)(C1n2c(C)nnc2CN1C(=O)OC(C)(C)C)OC12CC(O)C1C2 C(CC(C)(O)C(F)(F)F)NC(=O)NC(CC)(COC)C(=O)O.c1(C)ccccc1 C1(CNC(C2(COC)CCCC2)=O)C2CN(C(c3cc(O)no3)=O)CC12 C(=O)(CC1CCCNc2ccccc21)Nc1nc(C2CN(C)C3(C2)CCCC3)no1 C=CCC(C)(C)CCOC(=N)O.c12cccc(c1)N(C)CC(=O)C2 C(CC(CC)C(=O)NCCn1cc(CNC(c2sccc2COC)=O)nn1)=CC Cc1cc(O)nc(NC(=O)N(c2cccc(N(C)CC3(C)COC3)c2)C)n1 N1(CC(=O)N(CCOC)CCNC(c2[nH]cnc2C)=O)CSCCSC1 N1(C(c2ccc(SC)o2)=O)CC(NC(c2cnncc2O)=O)CC1CO C=CC1(C(N2CC3CCC2C(O)C3)=O)CCN(C(=O)CCCC2=CCCC2)CC1 CC1CC(NC(C2CC(C)(C(C)(C)C)C2)=O)CN1C(C1CC(C)(C)C1)=O c1(C(=O)NC2C(NC(C(COC)OC)=O)CCOC2)cnn2ccccc12 c1(CSCC(=O)N(CCC(C)NC(=O)C2=C(Cl)CCC2)C)ccc(F)cc1F c1(C(N2CC=CC(NC(c3c(C)nn[nH]3)=O)C2)=O)ccc2cn(C)nc2c1 CCS(=O)(=O)N(C(C)C(=O)N(CC(O)CNC(=O)CC1(CN(C)C)CCC1)C)C c1(NC(C(C)c2cc[nH]n2)=O)cn(C(C)C(=O)NCC2CC=CCC2)nn1 N1(C(c2cc(C)[nH]n2)=O)CC(C(=O)NCC(C)C(F)(F)F)OC(C)C1 c1(C(=O)NC23CN(C(C4(CC=C)CC=CC4)=O)C(CC2)C3)ccc(F)cc1C#N C1(=O)CC(C(F)(F)F)N1.c1(OCC(=O)N(CC(COCC)O)CC)ccccc1 c1(C(c2n(CCCOC)nnn2)NC2(C)CC2(C)C)cc(C#N)n(C)c1 Cc1c(C(F)(F)F)n[nH]c1C(=O)N(C)CC1CCN(C(C2(C)CC2C)=O)C1 c1(C(N(CC(C)NC(C2C(C)C2(F)F)=O)CC)=O)nnc2ccccc2n1 C1(C(N2C(C)CCC2CO)=O)CCCN(C(C)C(=O)N(C)C)CC1 Cc1cc(O)nc(C)c1C(=O)NCC(C)NC(C1(C)CCCCO1)=O Cc1sc(-c2ccco2)nc1C(=O)NC1CCCC(CNC(c2cc[nH]n2)=O)C1 C#Cc1ccc(CCCC(=O)NCCN(C)C(c2ccc(SCC)cc2)=O)cc1 N1(C(c2ccc(C)o2)=O)CC2CCC2(CC(=O)NCCC2CC2C)C1 c1(C(=O)NC2CN(C(CCC=C)=O)CC2(C)C)cc2ccccc2cc1F N1(C(C=Cc2c(C)ncs2)=O)CCC2(C(=O)NCC(F)(F)F)CCCC12 C(=O)(C(CC(C)C)NC(c1cnn(C(C)C)n1)=O)NC1(CCCC)CC1 C(=O)(CCCN=C1NS(=O)(=O)c2ccccc21)OC(c1ccccc1Cl)C(=O)OC C1(CC)CN(C(=O)C=Cc2ccoc2)CCN1C(=O)C(F)n1cccn1 C(C(CC)CCO)NCCCOC(C1(F)CC(C(=O)OCC)C1)=O C1(C)(C(=O)NCCCC#C)CC12CCN(C(C1CC13CCCC3)=O)CC2 C1(CNC(C(C)NC(C(CC)NC(C)=O)=O)=O)CCN(C)CC1 Cc1c(N(C)C)cccc1S(=O)(=O)N1CCC(OC(=O)NC2CCCC2)C1 c1(N(C(c2cccc(I)c2)C(=O)NCC(=O)OCC)CC)cccc(Cl)c1 c1(CNC(C2C(NC(C3ON=C(CC)C3)=O)COC2)=O)[nH]ccc(=O)c1O C#Cc1ccc(C(N2CCN(C(c3cnc(C#N)s3)=O)C(CCC)C2)=O)c(F)c1 c1(C(N2CCC(C(=O)Nc3cnc(OC)nc3)C2)=O)c(O)cccc1O C1(C(=O)NC(CCSCC)C)CC(NC(=O)Cc2cccc(F)c2)C1(C)C CCCC(F)C(=O)NCC1(CC(=O)N(CC(F)F)CCC)CC1 C1(CN)CC(CN2CCCC(C(N3CCN(C)CC3)=O)C2)CCO1 c1(-c2nnn(C)n2)ccc(-c2cccc(C(N3CCNCC3)C(N)=O)c2)cc1 C(=O)(C1Cc2ccccc21)NCC1C(C(=O)NC2(CC=C)CC2)CCCC1 C(CCN=c1nc2cccc(Br)c2c[nH]1)N(C(=O)Cn1nnc(C2CC2)n1)C N1(C(CC(C(C)C)C)=O)CCC2CCN(C(=O)CN(c3ncccn3)C)CC2C1 c1(C(C(=O)NC)N(CCCCCSC)C)cc(C(N)=O)sc1C C(c1c(C)coc1C)=CC(=O)N(C1CCN(C(c2cc(CC)ncc2)=O)CC1)C CC1=NN(C)C(=O)C1CC(=O)NC1CN(C(c2sncc2C)=O)CC1CO Cc1cc(=NC(=O)C2COCCN2Cc2sccc2Br)[nH]n1C c1(CN(CCC)CCNC(=O)CCC2CC2C)nsc2ccccc12 C1(O)(C(C(=O)NCCCCOC)F)CN(C(C2C=CCS2)=O)C1 N1(C(C2CC2F)=O)CC2CCCN(C(=O)CCc3nccs3)C2C1 C1(C(N2CC(NC(Cc3c(C)nc(C)s3)=O)C(C)C2)=O)CCOCC1(C)C c1(C(=O)NCC(C)N(C(=O)CCC2CC2(C)C)CC)ccc(C(C)C)nc1 CS(C)(=O)=NCCN=c1cccc(S(=O)(=O)NC2CCSC2)[nH]1 C1(NC(c2nc(C)c(C)o2)=O)CCN(CCOCC(C)C)CC1C Cc1cc(C(F)(F)C(=O)NCC2(CNC(C3SCCCS3)=O)CC2)cs1 N1(C(c2cnc(C)s2)=O)CCC(C)(CNC(c2ncccc2O)=O)C1 c1(CSc2cn(CC(O)CC3CC3)nn2)noc2c1CCCCC2 c1(-c2cc(OC)ncc2)cccc(F)c1CN1CCOCC(O)C1 N1(C(C(C)NC(=O)CN(C2CCC2)C)=O)CCCC(C)(C)C1C C1(NC(c2[nH]nc(OC)c2Cl)=O)CCCCC12CCCN(C(C1CC=CC1)=O)C2 C(=O)(C1c2c[nH]nc2CN1C(C1CC2(C1)CC21CC1)=O)NCc1ncn(C)c1 C(=O)(CC(=O)NCC1(C(=O)NCCOC(F)F)CCC1)OC C(=O)(C(CNC(=O)CCCCN(C)C)CC(C)C)NC(c1nc(C)on1)C C1(NC(CCN(C(CC(C)F)=O)CCCO)=O)CCCC1(C)C C(=O)(C1=CC(O)CCC1)NC1CCCC(NC(Cn2c(C)nnn2)=O)C1 CCCC(CC)C(=O)N(CC(C)(C)C(=O)NC1CCC(C2CC2)C1)C C1(NC(c2ccc(OC)c(Cl)n2)=O)C2CCC1CN(C(C1CCCCC1O)=O)C2 c1(CC)cc(C(N2CCC(OCC(=O)NC(C(O)CO)C3CC3)C2)=O)n[nH]1 c1(C(=O)NC2CCN(C(CSCCOC)=O)CC2O)ccc(F)c2ncccc12 N1(C(C2N(C)CC(O)C2)=O)CCC(C2CN(C(=O)CCc3nccn3C)C2)CC1 N1(C(c2ccc(CC)cc2N)=O)CCC2(CC1)CN(C(C1CCC(OC)C1)=O)C2 C1(C(N2CC(NC(=O)C=CC3CCCCC3)C(O)C2)=O)C2CCC(F)(F)C12 C1(C(=O)NCC2CCN(C(CCCOCC=C)=O)CC2C)CCc2nccn2C1 CC(=NO)c1cc(C(N2CCN(C(C3CCCC4CCCN34)=O)CC2)=O)cnc1O C12=c3c(n(C)nc3)=NC(=NCCN(C)C1)N2.S(=O)(=O)(CC)NCCCOC=C C1(=O)C(CCC)N1.C=CCCOCC(=O)NC1CC1CN(C(C)(C)C)C(C)=O Cc1n[nH]c(=NCC2CN(C(C3(Sc4ccccc4)CC3)=O)CCC2C)o1 C1(NC(Cc2n(C)nnc2)=O)C2CCN(C(c3ccc4c(c3)OCO4)=O)CCC12 C1(NC(c2cnc(C(C)C)[nH]2)=O)CC(OC)CN(C(c2sccc2C(C)=O)=O)C1 c1(C(N(C(CCNC(Cc2cc(C)nn2C)=O)C)C)=O)cccc(P(C)(C)=O)n1 C1(NCCC(C)(C)N(C)C(=O)OC(C)(C)C)C2CCC3(COC(=O)C13)O2 N1(C(=O)C(c2ccccc2)O)CCS(=O)CC1c1ccccc1 c1(NC(C2CCSC2)=O)cccc(-c2ncc(Br)cn2)c1 C1(CC)CC(N(C)N2CCCN(C(c3ccccc3)=O)CC2)C12CCCC2 C#CCC(CC(F)F)C(=O)N1CC(NC(=O)CCCC#CC)C(n2ccnn2)C1 Cc1cc(C)c2c(Cl)c(NC(=O)Cn3cc(C4C5CCCCC45)nn3)sc2c1 C(CC(C)NC(=O)OCc1ccccc1)(c1nnnn1C)NCC=C=C N1(C(Cc2c(C)n[nH]c2)=O)CCN(C(=O)CN2CCC(N(C)C)CC2)CC(O)C1 C1(C(N2CCC(CCNC(c3cn(C)c(O)n3)=O)C2)=O)OCC2CCCCC12 C#Cc1cc(F)c(C(=O)NCCC(O)CNC(=O)CCC(C)S(C)(=O)=O)c(F)c1 C(=O)(C(C(C)C)NC(c1ccccc1OCc1cccs1)=O)NCC(C)OC S(=O)(=O)(c1cccc(C(=O)NCCC(N2CC3CC3C2)=O)c1)N(C)C c1(C(=O)NC2CC3CN(C(C4(C)C=CCCC4)=O)C2C3)cnn2cccc(Cl)c12 c1(C(=O)NCC(c2ccc(F)c(Cl)c2)(C)C)cnc2c(cnn2C(C)(C)C)c1 C1(C(=O)NCC(C)(C)OCCNC(c2scc(OC)c2)=O)SC2C=CC1CC2 c1(OC)cc(Br)ccc1CNCC1CCCN(C(c2cc(Br)c[nH]2)=O)C1 c1(NC(=O)NC(CC(C)=O)C)c(F)cccc1Br CC1CCC(NC(=O)Cc2cncn2C)CN1C(=O)COc1cccc(C#N)c1 N1(C(CC2ON=C(CC)C2)=O)CC2(C1)CN(C(c1ccnc(C(F)(F)F)c1)=O)C2 C12(CC(N3CC(CNC(C4CSCC(=O)N4)=O)C3)=O)CCC(CC1)OC2 C1(CCNC(Cc2nc(C)[nH]n2)=O)C(C)CCCN1C(c1cnnc(O)c1)=O c1(OCC)c(F)c(C(N2CCN(C(=O)C(C)C)C3(CCC3)C2)=O)cc(F)c1F CCC(CC)CCC(=O)NC1CC1CNC(=O)CN(c1ncnc2[nH]cnc12)C C(c1ccc(F)cc1)=CC(=O)NCCN(C(c1ccnn1CCF)=O)C1CC1 N1(C(C2(CCNC(=O)CC(O)C3CCCC3)CCC2)=O)CC2C=CCC(C2)C1 C1(C(N(CC(CN(C(=O)CC2CC2(C)C)C)O)C)=O)CCCCN1CC(F)F c1(N2CC(C(C)NC(C3CCN(C4CC4)CC3)=O)OCC2)cnc(C#N)cn1 CN1Cc2ccccc2C1CNC(=O)NC1CCc2nncn2C1 c1(C(N2CCC(C(=O)NC3(COCC)CC3)C2)=O)ncc(N)cc1C N1(C(=O)Cc2csc(Br)c2)CCC2(CCCN(C(C3CCC4CC4CC3)=O)C2)C1 c1(CN(C(c2cnc(C3CCC3)s2)C(=O)NCCOC)C)ccc(C#N)cc1F CCC(CC)(CC)C(=O)NCC(O)CN(C)C(c1nccc2cc[nH]c12)=O c1(NC)ccc(C(=O)NC2CCC2NC(C2(c3ccc(F)cn3)CC2)=O)cc1 C(=O)(N1CCCc2nccn21)C12CC(NC(C3C(C)(C)COC3)=O)(C1)C2 C1(C#N)(C(N2CC(=C(CNC(C3C(=C)C3)=O)F)C2)=O)CCOC1 N1(CC(=O)NCCOCCN(C(CCN(C)CCO)=O)C)CCCNC1=O C=CCCN=C(NCCCOc1ccccc1)N1CCC(C2NC(=O)NC2=O)C1 C#Cc1c[nH]nc1C(N1CCC(N(C(=O)C=Cc2sccc2C)CCO)C1)=O C1(C(CN(C)C(C23CC(C2)C3)=O)=O)CCC(C(F)(F)F)CC1 Cc1ncc(C=CC(=O)NC2CCC(CNC(=O)Cc3ccnn3C)C2)c(O)n1 C1(NC(C2(CC#C)CCOC2)=O)CCN(C(c2sc(CCC)nc2C)=O)CC1C C1(C(=O)OC)CC1C1CCN(C(c2cccc3o[nH]c(=N)c23)=O)CC1 N1(C(CCCOC(C)=O)=O)CC(CNC(c2cn(C)cn2)=O)CC1C C1(C)(C(=O)NCC(CCNC(C2(CCCC)CCC2)=O)O)CC(C(C)C)=NO1 C=C(F)CN=C(NC1CC1C)NC1CCN(C(=O)C(CC)CC)CC1 c1(CNC2CCN(C(c3cc(C)c(O)cc3)=O)CC2F)cc(Br)cc(F)c1O C1(O)(CC(=O)NC(C(=O)OC)CO)CCN(C(=O)CCCc2sccc2C)CC1 c1(OC)cc(NC(=O)CC2CC3(C2)CN(Cc2ncco2)C3)cc(Br)n1 C(=O)(C1=CCC(C)(C)CC1)NC(CCOC)C(=O)NCc1cncn1C1CC1 C1(C(N(C2(C#C)CC2)C)=O)CN(C(=O)Cc2ccccc2F)CC12CCC2 c1(CC)cc(C)c(C(=O)NCCCNC(C2(CC(F)(F)F)CC2)=O)o1 C1(C(=O)NCC23C(CN(C(C4CCCCCC4)=O)C2)C3)CC2C(C1)C2(F)F n1(CC(=O)NC(C)C(CO)NC(C2(CCF)CCC2)=O)c(O)nc2ccccc12 C1(C(=O)NCC(N2CCCC2)C)CN(C(c2ccc3c(c2)CC3)=O)C2(CCC2)C1 N1(C(C2CCN(C(C)=O)CC2)=O)CCCC(N(C)C(c2ccc(C)cn2)=O)CC1 c1(C(=O)NC2CN(C(C3C(OC)C3)=O)CC2C)cc2sccc2[nH]1 N1(CC(C)NC(C2(COC)CC=CC2)=O)CCN(C(C2CC(O)(C#C)C2)=O)CC1 c1(NC(=O)NCCC(=O)NCCN(C(=O)Cc2cnccn2)C)cccnc1 c1(C(N(C2CCN(C(c3cncc(C)n3)=O)C2)CCC)=O)cn(C)cc1C Cn1c(=O)oc2c(C(N3CCN(C(C4CCC(C)(C)C4)=O)CC3)=O)cccc12 C#CCC(CC#C)C(=O)NC1CC(CNC(C2COC(=O)O2)=O)C1 Cn1nc(C(=O)NC2CCC(CNC(=O)CC3CSC3)C2)c2cc(F)ccc12 n1(CCC(=O)NCC(CC=C)NC(=O)CCC=CBr)cccnc1=O CCC(CNC(c1ccc(N(C)Cc2cc(C)no2)cc1)=O)C(C)(F)F C1(N(C(=O)C(F)C2CCOC2)CC)CCN(C(=O)CNC(=O)OC)CC1 c1(C(=O)NC(C2CN(C(=O)C(C)Sc3ccccc3)C2)C)ccc(CO)cc1 C1(C(N2C(C)(C)C(CNC(=O)C3=CCCOC3)CC2)=O)CCC2(CCOCC2)O1 C=CCCCC(C(=O)NOCC1CC1)NC(=O)CCC(=O)NC c1(C(=O)NC23C(CN(C(C4ON=C(CC)C4)=O)C2)C3)ccc(C)c(S(N)(=O)=O)c1 C(=O)(CC(C)C(F)F)N1CCCC(N(C(Cc2nnc(C)o2)=O)CCF)C1 c1(NC(C2CCC(CNC(C3CC4C=CC3C4)=O)CC2)=O)c(Br)ccc(F)c1F n1(CC)nnnc1C(C1(CSC)CC1)NCC1CC(C(=O)OC)C1 N1(C(C(C)CC#N)=O)CCC(N=[N+]=[N-])(C(=O)NCC2C(C)(C)C2(C)C)C1 C(=O)(C(CO)C(C)(C)C)N1C(C(C)C)C(NC(=O)CCc2cccnc2)CC1 Cn1cc(C(N2CCCCC2C(=O)NOCC2CCCO2)=O)ncc1=O CCC(C)CCCC(=O)NC1CCC(NC(=O)CC2=CCCC2)CC1 C=CCCC(O)CNC(c1ccn(CCNC(c2cnc(C)o2)=O)c1)=O C12(CNC(C(C=C)(C)O)=O)CCC(CN(C(c3cn(C)nc3O)=O)C1)C2 C(CC(C)(C)CC(=O)N(CC(=O)NCC1(CO)CCCO1)CC1CC1)OC C(=O)(CCC(C)(C)C(=O)NCCC1CCN(C(=O)Cn2nccn2)C1)OC Cc1ccc2sc(C(N3CC(C)CCC3CNC(C3(C4CC4)CC3)=O)=O)cc2c1 C1(C(C)NC(=O)C(F)=C2CCCC2)CCN(C(C2CC2c2cncn2C)=O)C1 N1(C(CSCC=C)=O)CCC(n2cc(CNC(C3(COC)CC=CC3)=O)nn2)C1 N1(C(C(C2CCOCC2)C)=O)CCC(NC(c2ccsc2C(F)F)=O)C1(C)C c1(CC(=O)N(CC(C)NC(C(C)OC)=O)CC)ccc(S(=O)(=O)N(C)C)s1 C1(C(=O)NCC(C=C)(C)C)CCCCCC1NC(=O)C(C)(C#N)CC c1(C(C(=O)NC2OCC3CCCC23)NC(C(CC)CC)=O)cc(C)cc(C)c1 C1(NC(CC(CC)O)=O)CCCC12CCN(C(C1CN=C3N=CNN3C1)=O)CC2 CC1CC(C(=O)Nc2ccccc2-c2ncc[nH]2)CCS1(=O)=O CCC(F)(C(=O)OC)C(=O)N1CCC(Cc2cn(-c3cccc(CO)c3)nn2)C1 CCCCC(C(=O)NC1CC(CNC(c2cc(C)ccc2O)=O)C1)ON=C(C)C N1(C(c2c(CC)non2)=O)CC2(C(=O)N(CC(C)(C)N(C)C)C)CC1CCO2 C1(NC(=O)CCc2ccccn2)CC2(C1)CN(C(=O)Cn1ncccc1=O)C2 C12CC3(C1)CC(C3)C(=O)N2.c1(-c2ccn(CC)n2)ccc(Cl)c(C(=O)OC)c1 N1(C(C(C)=CC)=O)CCCC(C2(NC(c3noc4c(F)cccc34)=O)CC2)C1 C1(CNC(C(CC)=CC)=O)(CNC(C2CCC(C(=O)OC)C2)=O)CCOCC1 C1(F)(CNC(c2cc(CC)sn2)=O)CCN(C(=O)C(C)C2CCCC2)CC1 CCC(C(=O)OC)C(=O)N1CCOCC1c1cn(Cc2ccc(F)cc2)nn1 C(=O)(C(F)C(F)(F)F)NC(CNC(C1CSCCS1)=O)CO C1(C(=O)NCC2C(NC(c3cc(Br)c[nH]3)=O)CCCC2)CC2(CCC2O)C1 CCC(C)(COC)C(=O)NC(C)CCc1ccco1 CN1CC=C(C(=O)N2C(CC(=O)NCc3noc(C(N)=O)n3)C3CCCC23)C1 N1(C(C(COC)O)=O)CCC2CCC(C1)N2C(C1(c2ncco2)CCC1)=O N1(C(C2(COC)COC2)=O)CCC(C(=O)NCC(C)C(C)(C)C)CC1 C(=O)(C(CCC1CC1)NC(=O)Cc1c(C)noc1C)NCC(C)SC C1(C(=O)NCC2CCN2C(=O)CCOc2ccc(F)cc2)CCC2(CCC2)CO1 C(=O)(CC(C)C(C)(C)C)NCC(C)N(C(CC(CC)CC)=O)C c1(N(C)C(=O)OC(C)(C)C)cc(CNC(=O)NCCC(F)(F)Cl)nn1C c1(OC)cc(C(=O)NC2CC(CNC(c3nncs3)=O)C2(C)C)ccc1F C1(C(=O)Nc2cccc(NC(CCCCC#N)=O)c2)CCC2(CC1)CC2(F)F C(=O)(C(C(C)(F)F)c1ccccc1)N(CCC(C)NC(C1CCCCC1)=O)C N1(C(C(C)(F)F)=O)CCC2(CCC(NC(C3CNC(=O)N3)=O)C2)CC1 c1(C(N(CC(C)O)CCNC(=O)Cc2cnsc2)=O)ccnc(OC2CC2)c1 CC(F)(F)C(F)C(=O)N1CC(O)CC1CC(=O)NCC1CCCOC1 N1(C(c2cc(CSC)no2)=O)CCCC(CO)(NC(=O)CCc2ncccn2)C1 C(=O)(C(C)(C)C(O)CC)N(CCCNC(c1nc(OCC)oc1)=O)C C1(NC(C(C)=C(C)C)=O)CCN(C(c2ccc(-c3ccccc3)nc2)=O)C(C)C1 C1(OCC(=O)NC2(CNC(c3c(C)con3)=O)CCC2)CCCCCC1 c1(C(N2C(CNC(CCOCC)=O)CC(F)C2)=O)cc(OC)cc(OCC)c1N c1(C(=O)NCC2(O)CCN(C(Cc3c(C)cco3)=O)C2)cc(C#N)oc1C CC(C)C(C(C)NC(=O)C(=O)NCc1ccc(F)cc1)NC(=O)CCCC#N n1(C2CC(N(CC3C(NC(=O)C=CBr)CCOC3)C)C2)ccc([N+](=O)[O-])n1 Cc1ccc(C(=O)NCC2CC2NC(c2cc(Cl)cc(F)c2N)=O)c([N+](=O)[O-])c1 Cc1c(O)nc2ccccc2c1C(N1CCCCC(N(C(=O)C(C)C)C)C1)=O CC(N=c1cc(Cl)c2cccnc2[nH]1)c1ccc2nc(O)[nH]c2c1 c1(C(=O)NCC(C)NC(c2cn(C)cn2)=O)cccc2oc(=N)[nH]c12 c1(NC)ccc(C(=O)NC2CCCN(C(=O)CCN3CCCCC3C)C2)nc1 Cc1cccc(NC(=O)CN(C(C)C(=O)N(C)C)C)c1 C(=O)(CS(C)(=O)=O)NC(C(=O)NCCOCC(=O)NC)c1ccoc1 c1(C(N2C(CNC(COc3cn(C)nc3)=O)CCC2)=O)cnn(C)c1C#N S(=O)(=O)(c1cccc(Br)c1F)N1C(CNC(c2c(OC)nccn2)=O)CCCC1 Cc1nc(Cl)[nH]c(=NC2CCCCC2NC(=O)CC(F)(F)C(F)F)c1Cl N1(C(C(c2ccn(C)n2)(C)C)=O)CC2(CC(NC(C3CC4C=CC3O4)=O)CO2)C1 C1(C(=O)Nc2c(OCC)nccc2)CC(O)CCN1C(=O)C(O)C(C)C c1(NCC(CCCC)NC(c2nnn(C(C)(C)C)n2)=O)ncn(C)c(=O)c1Br C=C(C)CN=C(NCC(c1cn(C)cn1)N1CCCC1)N1CCc2ncsc2C1 c1(CNC(C2C(NCc3c(C)ncs3)CCC2)=O)ccc(F)cc1Cl c1(NC(c2cc(OC)c(Cl)s2)=O)cccc(CS(C)(=O)=O)c1C C(N=C(NCC(=O)NCC1CCCCO1)NC1CCC1)C1N(C(C)C)CCC1 N1(C(c2cnc(C3CC3)s2)=O)CCC2C(CCCN2C(=O)CCC2CCCO2)C1 c1(C(N2CC(C)(NC(=O)CCNC(N)=O)C2)=O)ncccc1S(=O)(=O)N(C)C c1(C(N2C(CCC(=O)N(C3CC4CC4C3)C)CCC2)=O)ccc(O)cn1 CC(C)CCC(=O)C(=O)N1CCC1CNC(c1cccc(CF)c1)=O N1(Cc2cn(CCN(C(C(CC(C)C)(F)F)=O)C)nn2)CCC2(CCCOC2)C1 CS(=O)(=O)c1cc(C(N2CC3(CC(NC(=O)CCOCC4CC4)C3)C2)=O)cs1 N1(C(C2(C)COC2)=O)CCOC(CCNC(c2cccc(C(C)(C)C)c2)=O)C1 C1(C(=O)NCC(C2CCCC2)=O)CC=CC(n2cc(C3(O)CCCCC3)nn2)C1 C1(NC(=O)Cc2c(Cl)cccc2Cl)CCCN(C(=O)C=C2CCSCC2)CC1 C1(C(=O)NC(CN(C(C2(C#C)CC2)=O)C)Cc2ccccc2)CCOCC1C c1(C(=O)NCC(CN(C(C(N2CCNC2=O)C)=O)C)O)cc2sccc2s1 C1(C(=O)NCCC(C)CCNC(=O)C(C)(C)CC(F)F)CCCC2(CCC2)O1 C(C(=O)NCc1cccs1)(C1=NOC2CC12)N1C(C2(C)CC2)CCCC1 C1(CNC(=O)COCCF)CN(C(c2cncs2)=O)C2(CCC2)C1 c1(NC(NNC(=O)c2ccc(OC)s2)=O)c(C)nc2n1CCCC2 C(=O)(CC(CC)NC(=O)C=CCN1CCCC1)NC(COCC)C C(=O)(C(C)(C)C)NCCC(=O)NCC1C(NC(CC2CC(=C)C2)=O)C1 S(=O)(=O)(c1cccnc1Cl)N1C(C(N(CCOC)C)=O)CC(O)C1 c1(CN2C(C(N3CC4C(CO)C4C3)=O)CC(F)(F)C2)ccc2c(c1)OC(F)(F)O2 c1(N2CC3CC(=O)NC3CC2)nc(=NCc2cccnc2)[nH]c2ccsc12 c1(C(N2CCCC(NC(C(=O)NCC)=O)C2C)=O)cc(C)c(F)c(C)c1 c1(C(=O)NC2CC(CC(=O)NCC(CC)(C)O)C2)ccnc(NC)n1 C1(C(=O)NCCN2CCC(NC(c3ccsc3Cl)=O)CC2)CC2OC1C1CC21 N1(CC)CCOC(C(=O)NCC(CNC(c2ccnc(C(F)F)c2)=O)CO)C1 C(=O)(C(O)(CN(C)C)C(F)(F)F)N1CCC(NC(CC(CC)CC)=O)(COC)C1 c1(SC)cc(C)c(C(=O)NCC(C2(O)CCN(C(=O)CCc3cnoc3)C2)C)o1 C1(CC(=O)NCCOCCCN(C(CCNC(=O)OCC)=O)C)CCCOC1 c1(C(N2CC(O)(CCNC(C(P(C)(C)=O)O)=O)C2)=O)c(F)ccc(F)c1F c1(C(=O)NC(C(C)NC(CS(=O)(=O)NCC)=O)C)cccc(C)c1N CC1CCN(CC(=O)NCc2c[nH]nc2C2CCN(C(=O)CSC3CC3)C2)CC1 C1(NC(Cn2nnc(C)n2)=O)CC(C2CCN(C(c3ccc(F)cc3O)=O)C2)C1 Cc1[nH]nc2ncnc(N3CCC(CF)(NC(=O)C(C)C4CC4)C3)c12 c1(C(=O)NCC(C2CCOC2)NC(C(CC)(F)F)=O)cnc2c(c1)COCC2 c1(C(C(N2CCN(C3CCN(C(C(C)=CC)=O)C3)CC2)=O)O)ccc(Cl)cc1F C1(OCCNC(C(=O)OC)C(C)c2ccccc2)CCN(S(=O)(=O)N(C)C)CC1 C1(NC(CCOC)=O)COCC1n1cc(C2(O)CCCC2)nn1 C(CN=c1[nH]c(=NCc2ccc(C3CC3)cc2Cl)[nH]c2c1CCC2)SC(F)(F)F c1(C(N2CCCC(CN(C(c3cc(OC)ncc3)=O)C)C2)=O)cccc(C)c1C c1(C(CCOC)NC(C2CCNC2c2ccccc2)=O)ccccc1C N(C1CC2(CCCC2)c2ccccc21)C(C(=O)NC1CCCN(CCO)C1=O)=O c1(CC(N2CCC3CCC23CNCCC(C)(F)F)=O)cccc2ncccc12 c1(C(N(CC(C)NC(c2cc(CC)oc2C)=O)C)=O)cc(F)cc2nccnc12 C1(CC(N2CC(=C(CNC(C3CCCC3(F)F)=O)F)C2)=O)CC2(CCC2)C1 c1(C(=O)NCC2(CNC(C34CCCC(CO3)C4)=O)CC2)cnc2nccn2c1 CCCCC(O)C(=O)NC12CC(C1)N(C(=O)C(C)OCCN(C)C)C2 c1(C2(C(=O)NCCCC(C)(C)C)CC2)cccc(Br)c1F CN1CCN(C(=O)Cn2cc(C3COCCN3)nn2)C1=O CC1(NC(C2CCC(NC(=O)C=Cc3cncs3)CC2)=O)CCSCC1 c1(C(N(CC(CCC)C)C)=O)oc(CNC(c2ccncc2)=O)nc1C C(=O)(C(CCC1CCC1)NC(C1CC=CCC1)=O)N(CC(C)C)C(C)C C(=O)(C(Cc1ccc(O)cc1)C(F)(F)F)NCC(C)NC(CC=C=C)=O N1(C(Cn2c(C)ncc2)=O)CCC(NC(c2ccnc(CO)c2)=O)C(CO)C1 Cc1ccc(CCNC(C2C3CCC2(c2nccs2)C3)=O)c(C)c1 N1(C(C#CC(C)C)=O)CC2CCC(C(=O)NCCCC3CC3C)(C2)C1 C(=O)(CC(CC#C)NC(c1oc(C)nc1CC)=O)N(CCCC#C)C CS(=O)c1cccc(C(=O)NC2COCCC2NC(c2nocc2C2CC2)=O)c1 C1(C(=O)NCC(CCNC(c2occ3c2CCCC3)=O)O)COC2CCCCC12 C#Cc1cncc(C(N2CCN(C(=O)C(C)OCC3CCCO3)C(C)C2)=O)c1 N1(C(C(C)OCC=C)=O)CCC2CCCC(C1)N2C(=O)CSc1ccccc1 C1(C)(CNC(C(C2CN(C(c3n(C)ccn3)=O)C2)O)=O)CC(C)(C)C1 c1(C(N2CC(CCCCNC(c3c(C)scc3)=O)C2)=O)cncc(C(=O)N(C)C)c1 c1(SCC(=O)NC(C2OCCN(C(CC(C)OC)=O)C2)C)ccc2c(c1)CCC2 C1(NC(CC(=O)N(C)C)=O)CC2CC1N(C(=O)CCc1nncs1)C2 C(=O)(C(C)C(O)C(C)C)NCc1ccc(C(N(CCC)C2CC2)=O)nc1 CC1CC(CNC(=O)COc2ccccn2)CCS1 C1(C(=O)NCC2CC(OC)CN2C(C2CCCC2(C)C)=O)CS(=O)(=O)CC12CC2 C1(C(N(CC(COC)C)C)=O)(CNC(c2cnc[nH]c2=N)=O)CC12CCC2 Cc1cccc2[nH]cc(CC(N3CC(NC(=O)CCC(C)C)C4CC34)=O)c12 C12(NC(COC(=N)O)=O)CCCC1CN(C(C1(C(=O)C3CC3)CCC1)=O)C2 C(=O)(C(C)(C)C(C)(C)O)N1CC(CC(C(N2CCC(NC(=O)OC)C2)=O)F)C1 C1(C2CCCO2)(C(=O)NCC#CCNC(c2cccc(C#C)c2Cl)=O)CCCO1 c1(-n2c(-c3csc(CO)n3)nc(CCCCC)n2)cc(C)nc(C)c1 C1(C(C)(C)NC(C(C2CCC2)OCC)=O)CCN(C(=O)CCc2ncc(C)[nH]2)C1 Cc1cccc(C(N2CC(O)(C(C)NC(C3CCN3S(C)(=O)=O)=O)C2)=O)c1C C12(C(=O)NCC3(F)CC(CNC(=O)Cc4csnn4)C3)CC(C(F)(F)F)(CO1)C2 c1(OC)c(Br)cc(CC(=O)Oc2cc(C(N)=O)cc(Cl)c2)cc1Br c1(C(N2CCN(C(C(C)(C)C)=O)CC2CC(F)F)=O)ncn2c1CCCC2 C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)N(C1CCN(C(=O)C=C2CCC2)C1)CC N1(C(c2scc(C)c2C)=O)CC(CC(=O)NC2CC(C)(O)C2)CC1(C)C c1(CC)[nH]c(=N)sc1C(=O)NCC1(CNC(c2cnc(C)nc2)=O)CC12CCC2 c1(CC2CCN(C(=O)CCC3CCCOC3)CC2)ccc(F)c(F)c1 C=C(C)CCC(=O)NC1CCCC1N1CCN(C(C2CC3CC3N2C)=O)CC1 N1(C(CN(C)C(c2ccsc2)=O)=O)CC2(CCCN(C(=O)CC3CNC(=O)C3)C2)C1 C=CCN=C(NCC1COCCN1CC)N1CCCC(C)(F)C1 CC(C)C(C)(CNC(=O)CCC(F)F)NC(c1ccnc(O)c1)=O N1(C(C2N(C(C)=O)C(=O)CC2)=O)CCC2(CC1)CN(C(C1(C#N)CC1)=O)C2 N1(CCNC(CC(C)NC(C=C(C)C2CC2)=O)=O)CCOCC1=O N1(C(c2ccc(C)cc2)=O)CCC2(CCCC2C(=O)Nc2ccc(C#N)cc2)C1 CC(C)C(O)C(=O)NC1CCN(CCNC(c2cnc(C3CCCO3)s2)=O)CC1 Cc1cc(C(=O)NC(CNC(c2nscc2Br)=O)C2CC2)nc(O)c1 C1(CNC(CN(C2CCSC2)C)=O)CC2(CCC2)CN1C(C1CC2(CSC2)C1)=O C1(CC)CCN(C(C2CCCC(=O)C2)=O)C(C(N2CCC2COC)=O)C1 C#CC12CCC(C(N3CC(CNC(c4scc(C)c4Cl)=O)C3)=O)(CC1)CC2 Cc1cc(P(C)(C)=O)oc1C(=O)NC(c1ccc(F)c(Br)c1)CO C1(C(N2CCN(C3CN(C(CCC4CC(OC)C4)=O)C3)CC2)=O)CCCCCCC1 C(c1ccc(SC)cc1)=CC(N1C2C(CNC(C(C)N(CC)CC)=O)C(C2)C1)=O N1(C(C2(C(C)C)CCC2)=O)CC(C(=O)NC2CCN(C)C(=O)C2)CC(C)(C)C1 c1(N2CC3(C(C(=O)Nc4cnc(C)nc4)C3)C2)ncnc2cccnc12 CC1C(=O)CCC1CC(=O)NC(C1CCN(C(C2C=CC=CC=C2)=O)CC1)C CCCC(CNC(c1oc(CNC(c2[nH]ccc2C2CC2)=O)cc1C)=O)CCO C(CC(C(C)C)NC(=O)C(CNC(=O)COCCCCC)CC1CC1)OC C1(CNC(C2(F)C(C)C2)=O)COCC2(CCN(C(=O)CC3CC=CC3)CC2)O1 C1(CNC(C2(OCC)CCC2)=O)CCC2CN(C(C3CCC4(CCC4)C3)=O)CC12 CC1=NOC(C(=O)NCC(O)CCNC(=O)COC2(C)CCCC2)C1C C1(=O)C(CNC(C)=O)NC(=O)N(CC)CCN1.c1(OC(C)(C)C)nnsc1N CCCCCC(=O)N1CC=CC1C(N1CCC(C(=O)NCc2ccsc2)CC1)=O c1(OCC)nc(NC(C)(C)CCNC(=O)C(C2CCC(=O)N2)C)ncc1C O=C1OC(C(=O)Nc2cccc(F)c2)Cc2cc(-c3nn[nH]n3)ccc21 C(CCC)(C(=O)N1CCC(=CCNC(C2(n3cnnn3)CC2)=O)CC1)=CCC c1(CC(N2CCC(NC(CC(C)SC)=O)(CF)C2)=O)ccc(Cl)c2cccnc12 C(=O)(C#CC1CCCCC1)N1C(CNC(=O)C=CC2CCOCC2)CCCC1 C12(CNC(CNC=O)=O)CCC(CC1NC(=O)CCn1cnccc1=O)C2 C(CCCCC(=O)NCc1cccc(C(=O)N(C2(c3cc[nH]n3)CC2)C)n1)SC CC1CC(C(=O)NCC(C)N(C)C)N(C(=O)CCCn2cncn2)C1 C1(NC(COCCCCC)=O)CCN(C(c2cnn3c2CCCC3)=O)CC(O)C1 C1(O)(CC(N2C(C(C)NC(c3csc(Br)n3)=O)CCC2)=O)CCCCC1 Cc1cc(CCCC(=O)NCCC2CCN(C(=O)C(C)N(C)C)C2)on1 c1(C(N2C(C)(CNC(=O)C(O)CF)CCC2)=O)ccc(F)c2ccccc12 C1(CCC(=O)NCc2cc[nH]c2C(=O)NCCCN2CCC2)CCCOC1 CC(C)(C(=O)NCc1ncco1)C1=CCN(C(c2ccc([N+](=O)[O-])o2)=O)C1 C=CCCC(C)(C)C(=O)NCC1C=CC(NC(=O)CCOCC2CCCO2)C1 c1(C(N2CC(NC(CCCOCC)=O)C(C)C2)=O)csc2c1CCCC2 Cc1cc(C)c(C(=O)NCC(C)(O)CNC(=O)C(C)N(C)C)c(O)c1 c1(C(=O)NC(C(CO)NC(CC2CCN(CC)C2)=O)C)cccc(OC(F)F)c1 Cc1cnc(NCCCC(C)CO)c(S(=O)(=O)NCC2CC(=C3CC3)C2)c1 c1(CN(C(CCN(C(=O)C(O)C=C)CC#C)=O)C)cccc(C)c1 c1(N2CC(CN(C)C(c3csnc3Cl)=O)OCC2)ncc([N+](=O)[O-])cc1C(N)=O CCCC(C(=O)N1CC2CC1C2CNC(=O)C(F)=C(C)C)NC(=O)OC(C)(C)C c1(C(=O)NNC(=O)C2CN(C3CCOCC3)C2)nccc2c(Cl)cccc12 C(=O)(C(C(C)(C)O)NC(=O)C(C)N(C)C)N(C1CC(C#N)C1)CC#C N1(CC(=O)NCC2C=CCN2C(C2CC2(F)F)=O)CCCC2(CC2)S1(=O)=O N1(C(C(C#N)C2CC2)=O)CCC(O)(CNC(c2ccc(OCCF)cn2)=O)C1 c1(OC)ccc(C(N2CCN(C(=O)NC(=O)C(Cl)(Cl)Cl)C(C)C2)=O)c(C)c1 C1(C(=O)Nc2cccc(C(N)=O)c2)CC12CCN(C(=O)CC1CCNC1)CC2 C1(CNC(CSCC#C)=O)CN(C(c2cccc(C(=O)N(C)C)c2)=O)CCC1C N1(c2ncc(C)c(C)n2)CC2CCCN(C(c3cccc(C(C)C)n3)=O)C2C1 N1(C(c2n(COC)ncc2)=O)CCC(F)(C(=O)NCC(c2ccccn2)O)CC1 N1(C(C=Cc2c(C)ncs2)=O)CCCC(NC(C2(O)CC2)=O)C1C C=C(CC(=O)OC)C(=O)OCC(O)C(C)C c1(C(=O)NCC2(NC(c3c(C)c[nH]n3)=O)CCCCC2)cc([N+](=O)[O-])nn1C C1(CC(=O)NC)CCN(C(=NCCC2CCOC2C)NCCCF)CC1 CCC(C)(C)CC(=O)NCC(C)(C(C)C)NC(=O)Cc1ncc(Cl)s1 C(CC(C)C)(C(=O)NCCC#N)N1CCC(c2cc(C)no2)CC1 c1(C(=O)NCC(C)(CNC(C2(CO)CCOC2)=O)OC)cc(C)c(C)c(C)c1 N1(C(CCCc2onc(C)n2)=O)CC2CC1CN2C(c1[nH]nnc1C(F)F)=O c1(CC(=O)NC(CCCNC(C2CC(C)C2)=O)C)cccc([N+](=O)[O-])c1 c1(OC)ccnc(OC)c1S(=O)(=O)N1CCC(S(N)(=O)=O)CC1 c1(C(=O)NC2CN(C(CCOC(C)=O)=O)CC(O)C2)[nH]c2ccccc2c1Cl c1(C(=O)NC2C3OCC(NC(CS(CC)=O)=O)(C3)C2)cc(S(N)(=O)=O)c[nH]1 C1(C(N2C(CNC(=O)CC(O)C3CCCC3)CCC2)=O)CCc2cncn2C1 C1(F)(CNC(C2(C)C=CCC2)=O)CCCN(C(C2CC3(C2)CC(O)C3)=O)C1 N1(C(C2N(C(C)=O)CCCC2)=O)CCC(NC(=O)CCSCC(C)C)C(F)C1 C1(NC(C2C=CCC2)=O)CCC2(CC1)CN(C(C13CCCC1C3(F)F)=O)CCO2 N1(C(COCCC)=O)CCC(C)N(C(=O)CC(O)C(C)CC)CC1 c1(C2CCN(C(C(=O)NC(c3nncn3C)C)=O)C2)ccccc1Cl N1(C(C(F)=C(C)C)=O)CC(NC(c2ccc(CN3CCOCC3)cc2)=O)C(F)C1 C1(C(=O)NCC2(NC(c3ccc(CO)cn3)=O)CC2)CN2CCC1C2 C1(C(=O)NC2C(CN=[N+]=[N-])CN(C(c3cnc(Cl)[nH]3)=O)CC2)CC1C1CC(F)(F)C1 C12CCCC1NC2.C(=O)(C(F)(F)F)NC1C(NC(C)=O)C1 c1(C(=O)NC2(CNC(CCOC)=O)CCCCCC2)cc(C)cc([N+](=O)[O-])c1 C1(NC(c2c(C)nco2)=O)CC(O)CN(C(=O)CCOCC2CC2)C1 c1(CO)cccc(Sc2cc(C3CCOCC3)on2)c1.c1(S)nnnn1C1CC1 c1(C(=O)NCC2CN(C(C(C)(C)OCC)=O)CC2C)c[nH]c2cc(F)ccc12 N1(C(C(=O)NC2CCC2)c2ccsn2)CCOC(C2CCOC2)C1 Cc1cc(C(=O)NC2COCCC2NC(C2CC2C)=O)nn1-c1cccc(Cl)c1 CCC(CCCC(=O)N1CC(C)=CC(C)C1)NC(c1cn(CC)nn1)=O Cc1cc(C)cc(C=CC(=O)NC(C)C(C(C)C)NC(c2nnc(S)n2C)=O)c1 C1(C(=O)NCCN(C)C(c2ncccc2N)=O)CC2CCC(C1)S2(=O)=O c1(C(=O)NCc2nc(CNC(=O)C=C3CC3)nc(O)c2)cnn2cc[nH]c(=O)c12 c1(C(=O)NCCCCCCN(C(C(CC#C)C2CC2)=O)C)cc([N+](=O)[O-])c(C)s1 C#CCC(C)C(=O)N1CC(N2CC(NC(=O)CCc3c(C)n[nH]c3C)CC2=O)C1 C1(N(C(C2N(CCC)CCC2)=O)C)CCC(CNC(c2ncccc2Cl)=O)CC1 c1(C(N(C2CCN(Cc3ccn(C)n3)C2)CC)=O)c(F)cccc1F C1(CCNC(CN2CC(=O)NC2=O)=O)CC2CCC(C1)N2C(C1(Cl)CC1)=O N1(C(c2c(CC)c[nH]c2)=O)CC(C(=O)N(C)CCc2cccs2)CC(C)C1 CCC(C)(C(=O)NCCC1CCCCN1C(=O)COCc1ccncc1)C(F)F CONC(=O)C(=O)N1CC(=O)CC1C(=O)NCc1c(F)cncc1F C1(OC)CCC2(CCN(C(C3CC=CCC3)C(=O)Nc3c(C)cccc3C)C2)C1 S(=O)(=O)(c1cccc(Br)n1)N1CC(F)(C(=O)Nc2cncc(Br)c2Cl)C1 N1(C(C(C)C2CCC2)=O)CC(NC(c2ccn(C)c2)=O)CC12CCC2 C(N=c1[nH]cncc1OC)C1C(NC(CNc2ccc(C#C)cc2)=O)CCCC1 CCC(CCCC(=O)NC1(c2ncc[nH]2)CC1)NC(=O)C=CC1CCOC1 c1(C(N2CCC(F)(C(=O)NCC=CCCC)CC2)=O)ccc2c[nH]nc2c1 C1(CNC(=O)CCN(CCCO)C(=O)CNC=O)CCC(=O)O1 C1(CNC(c2sc(C(=O)OC)c(N)c2)=O)CN(C)CCN1C(=O)C(C)OCC(C)C c1(COC(c2cc(OCC)c(Br)cc2)=O)c(C)nc(C(C)CC)nc1C C(=O)(C(F)CC1CCC1)N(C1(CC(=O)N(C2CCCOC2)CC)CC1)C C(=O)(C1(C)CCn2c(C)nnc21)NCC(CN(C(C(C=C)O)=O)C)(C)C N1(Cc2ccc(OC)nc2)CCC2CN(C(c3cccnc3)=O)CCC12 C1(C(C(=O)NCCCOCCC(=O)N(CC(COC)O)C)C)CCC(=O)N1 c1(-c2n(CCC#C)c(N3CCC(OCCF)C3)nn2)cnn2c1CCCC2C Cn1ccc(C(N2CCN(CCNC(=O)C(C)(C)CCl)CC2)=O)c1C1CNC1 CC1CC(NC(=O)Cn2[nH]cnc2=N)CN(C(C2(N(C)C)CCCCC2)=O)C1 C(c1cccc(Cl)c1)=CC(=O)NC(CC)CNC(=O)CCC(=O)NC n1(CC(=O)NCC(CC)NC(=O)C(C)OC(C)=O)cc(C(=O)O)cn1 N1(C(C2CCC(=C)CC2)=O)CC2(CNC(=O)C(CC)C(F)(F)F)CC(F)(C1)C2 c1(C(=O)NCCOCCNC(CCCCN(C)C)=O)cnc(O)c2ncccc12 N1(C(CCOC)=O)CC2CCC(C1)N(C(c1ccon1)=O)C2 C(=O)(C(CNC(=O)CCC1CC1C)CC(C)C)N(CCCO)CC c1(CC)cc(C)ccc1NC(C1CCCN(C(c2cnsc2C)=O)C1)=O CCCCC(CC)C(=O)N1CCCC1C(C)NC(c1ncccc1Cl)=O S(=O)(=O)(c1ccc(SCc2cccc3c2CCC3)cc1F)C(=O)O CC12CCC(C(=O)NCC3(CNC(c4[nH]ccc4C4CC4)=O)CC3)(C1)OC2 N1(C(C(CC)COC)=O)CCC2(CCC2)C(NC(c2cccc(CF)c2)=O)C1 CC(CN(C)C)C(=O)NC1CC(CNC(c2cnc(C3CCCO3)s2)=O)C1 c1(CC)ccc(C(=O)NC(CO)CCCCNC(C2CC(C3CC3)C2)=O)c(C)c1 C(=O)(CC(C)(C)COC)N(C1CCCN(C(=O)CCCCc2cnc[nH]2)C1)CC Cc1cn2nc(C(N3CCC(NC(=O)C=Cc4ncc[nH]4)CC3)=O)cc(C)c2n1 CC(C)C(C(=O)NCc1cscn1)NC(C1CN(C)C1)=O c1(OCC)nc(C)c(C(=O)NC2CCN(C(=O)CCC(C)OCC)C2C)s1 C(CC)(CC)(CCNC(=O)C(CC)Oc1cccc(Cl)c1)NC(C(F)=CCC)=O N1(C(C2C(C)=C2)=O)CCC(N(C(=O)CC2CC2)C)C1 c1(C(=O)NC(C(C)C)CO)ccc2c(c1)N(C)C(=O)CO2 C(N=c1cc[nH]c(C(C)C)n1)C1(c2c(C)cccc2)CCC1 N#Cc1nc(Cl)ccc1NC(C1CC(F)CN1C(=O)CCN1CCCCC1)=O C1(C(N2CCCC(O)CC2)=O)CCN(C(=O)C2(C3CC3)CCCC2)O1 C(C(C)C(=O)OC)SC.C1(=O)C(=O)NCCOCCN1 c1(C(N(C)CC2(CNC(C3(OC)CC3)=O)CC2)=O)ccc2cncn2c1 c1(OC)cccc(F)c1C(N1C(C(=O)Nc2cc(Cl)cc(Cl)n2)CC2CC12)=O C(=O)(C1Cc2ccccc21)NCC1OCCN(C(C2(S(N)(=O)=O)CCCC2)=O)C1 O=C1CC(C(=O)NC2(CO)CCN(C(C3CN(C4CCCCC4)C3)=O)C2)CN1O Cc1nc(C(N2CCC=C(C(=O)N(C)CP(C)(C)=O)C2)=O)ccc1C#N c1(CC(=O)NCCCN(C(=O)Cc2csc(S)n2)CCO)cccnc1 N1(C(C(C)CC2CCCC2)=O)CCN(C(c2scnc2C2CC2)=O)CC1CO C1(NC(C2(C3CCCC3)CCC2)=O)CC1C1CCCN(C(C2CCCCO2)=O)C1 c1(C(=O)NC(CNC(c2[nH]cc(C)c2C)=O)C(C)C)nnc(O)nc1O c1(C(c2noc(C(N3CCCC3)C)n2)OC)ccccc1Cl CC(C)CC(C(=O)N(C)CCNC(c1ccc(-c2ccncc2)cc1F)=O)C(N)=O CC1OCCC1CC(=O)NCC(=O)NCC1CCCS1 c1(SC)ccc(O)c(C(=O)NC(C2CN(C(c3n[nH]c(C)c3C)=O)C2)C)c1 Cc1cc(Cl)cc(C)c1C(N1C2CCC1C(CNC(=O)CC1CCCOC1)C2)=O c1(CCNC(N(CC(C)O)C(C)CO)=O)ccc2cnn(C)c2c1 N1(C(C(CCC)C)=O)CCC(NC(=O)CNC(=O)Cc2cccc(F)c2)C1(C)C Nc1cc(C(N2CCCCCC2CNC(=O)C=C2CCOCC2)=O)cc(Cl)n1 C(=O)(CCCC(CC)CC)N1CCCC(C(=O)NC(CCC)CCO)(CC)C1 c1(C(N2C(CO)CC(NC(c3cnc[nH]3)=O)C2)=O)ccc([N+](=O)[O-])[nH]1 c1(OC)nc(C)ncc1C(=O)NC1CC2CCC1(CNC(c1cc(Cl)no1)=O)C2 C1(CC)CCN(C(=O)C(CSC)OC)C1C(=O)Nc1cccnc1 c1(C(C(=O)N2CC(CNC(C(=O)NCC)=O)C2)(C)C)ccc(Cl)c(Cl)c1 C1(C(=O)NC2(CO)CN(C(=O)C(c3ccc(C)cc3)C)C2)(N)CCCCC1.CC C1(NC(CN(CCC)C)=O)CC2(CCC(CNC(C3CC=CC3)=O)CC2)C1 c1(OCC)nc(N(CC(C)CNC(C2CCCN2CC)=O)C)ncc1C Cc1cnc(C)c(C(=O)NCCC2CN(C(=O)COC3CCOCC3)CCO2)c1 C(=O)(CCC(CF)CF)NC(C(=O)N(C)Cc1snc(C)n1)(C)C1CCC1 c1(CN(CC(=O)N(CCNC(c2cn(CC)nn2)=O)C)C)cccc(C#N)c1 N#Cc1cccc(OCC(=O)NCCN(CCO)CC(=O)C=Cc2ccco2)c1 c1(C(N2CC(C)C(CNC(=O)CN3CCOCC3)C2)=O)cc(C(N)=O)cc(F)c1 N1(C(C(CC=C)C)=O)CCOCC2(COCCN2c2ncnc(=N)[nH]2)C1 n1(CC(=O)NC2(CCNC(CCC)=O)CC2)ccc(O)nc1=O C1(C(=O)NC(c2ccccc2)C#C)CC(C(=O)O)N(C(=O)OC(C)(C)C)C1 CC1CCCC(C)N(C(C2CC23CC(NC(C2C4(CC4)C24CC4)=O)C3)=O)C1 c1(OC)ccc(C(c2nnnn2C2CCOCC2)NCC2COC(=O)O2)c(C)c1 C1(C(=O)NC2CCC(F)(CNC(c3cnn(C)n3)=O)C2)CCC(=C(F)F)CC1 C#CCC(CC(=O)NC1(CC(=O)OC)CC1)NC(=O)C(C)(C)C1CCCO1 N1(C(C(CCCCC)O)=O)CCCC12CCC(NC(=O)C=C1CCC1)CC2 CN1N=CC(CC(=O)NCC2CC(C(=O)NC3CCCC(CO)C3)CO2)C1=O Cc1cc(C#N)sc1C(N1CCC(N(C(=O)C(c2ccccc2)F)C)C1)=O C(=O)(C1CCCc2nncn21)N1CC2(CN(C(c3cccc(=S)n3O)=O)C2)C1 c1(OC)ccc(C(=O)NC(CNC(c2csnc2C)=O)C2CC2)c(F)n1 N1(C(C(C)=CC2CC2)=O)CC(CNC(c2nccnc2N)=O)C2(CC2)C1 CC1(C)OCC2CC12C(N1CC(Nc2nccc(C#N)n2)C1)=O Cc1nc(N)cnc1C(=O)NCC1CCCC(CNC(c2csc(O)n2)=O)C1 N1(C(C(C#N)=CC(C)C)=O)CCC(C)(C)C(CNC(C2CCOC(C)C2)=O)C1 C#CCC(CC#C)C(=O)N1C2CCC1CC(N(C)C(C1CC(F)C(=O)N1)=O)C2 N1(C(c2n(C(C)C)ccn2)=O)CC(C(=O)NCC(O)CO)CC(C)C1 CC1(C#CC(=O)N2CC(O)CCC2C(=O)NCCn2ccnn2)COC1 CC(C(=O)NCC1CCC1C(N1CC(O)C1)=O)c1cc[nH]n1 c1(N2CCN(c3c([N+](=O)[O-])cccc3)CC2)ccc([N+](=O)[O-])cc1Cl N1(C(C(C2CCCC2)OC)=O)CC(NC(c2cc(Cl)ns2)=O)C(F)C1 N1(C(Cc2ccc(OC)cc2)=O)CCC(NC(=O)C=C(C)C(C)C)C(C)(C)C1 C1(CC)CCN(C(C2(NC(c3cnc(Cl)s3)=O)CSC2)=O)C1 c1(C(N2CCC(NC(CCC=C(C)C)=O)C2(C)C)=O)cc(O)cc(C#N)c1 C#CC(C1CCc2ccccc21)NC(=NCC=C)NCC(=C1CCOCC1)F C1(C(=O)NC(CN(C(c2ncncc2Cl)=O)CC)C)C2CN(CC(F)(F)F)CC12 C1(C(=O)NCC(COC(C)C)O)C2CCN(C(=O)Cn3ncnn3)CC12 C12(C(=O)NC3C(C)OCC3)CC(CO1)N(C(=O)CCCC1CC1C)C2 c1(N2CCC(C)C(F)(F)C2)nccc(=NC(C)c2ccc3c(c2)CCCC3)[nH]1 c1(C(=O)NC(C(c2ccccc2)NC(C=NOC)=O)C)ccc2nccnc2n1 c1(C(N2CCC(C3N(C(c4c(OC)scc4)=O)CCC3)C2)=O)cc(Br)n(C)c1 Cc1c(Br)ccc(O)c1C(=O)NCC1CC1NC(=O)CC(C)C(F)F C(=O)(C(F)(F)C(F)F)N1C(C(=O)NC2CC(Cl)(Cl)C2)CC2CC21 n1(CC)cnc2[nH]c(=NC(C)c3cncs3)nc(N3CCOC(CF)C3)c12 O=C(C1=CC2(CCOCC2)C1)N1CC2(CCN(Cc3ncoc3C3CC3)C2)C1 C1(COC)CN(C(c2cc(N)ccn2)=O)CCN1C(c1sncc1C)=O c1(NC2(c3n(CC(=C)C)nnn3)CC(CCCC)C2)cnc2ncccc2c1 c1(N2CC(C)C(NC(C3CCS(=O)(=O)C3)=O)C2)nc2c(cc1C#N)CCC2 C1(C(c2nnnn2CCCSC)NCCC=C=CC)COCCN1CC N1(C(C(CC)=CC)=O)CCC(O)(C(C)CNC(C2CN(C(N)=O)C2)=O)C1 C1(C(N2CCC(NC(=O)CCN3CCCCC3=O)(CO)C2)=O)CC2OC1C1CC21 C1(CC)CN(C(C2CCS(=O)(=O)C2)=O)CCN1C(C1CN(C(N)=O)C1)=O N1(C(C(C)CC2CCC2)=O)CCC2(CCCN2c2ncnc(=N)[nH]2)C1 C12(C(=O)NCC3CN(C(c4c(C)ncs4)=O)C3)CCC(CC1)C(C)(C)O2 c1(C(=O)NCC2N(C(c3c(C)nc[nH]3)=O)CC(O)C2)ccc2ncncc2c1 C1(O)(C(C)NC(=O)C2=CCSC2)CCN(C(c2cc(C3CCOC3)[nH]n2)=O)CC1 CCCC(CC)C(=O)N1CCN(C(c2cc(F)ccc2NC)=O)CC1C C#CCCN=C(NCC1CC2CCC2C1)NCC(c1ccncc1)O c1(C(N2CC(CC)C(NC(=O)C(C)SC)C2)=O)cc(C)c2n[nH]cc2c1 C(=O)(C1=C(Cl)CCCC1)NCC(C)CN(C(=O)C(C)(C)Cc1cnn[nH]1)C Cc1[nH]nc(C(=O)NCC(C)(C2CC2)NC(C2CC2c2ccn(C)n2)=O)c1C Cc1c(C(=O)NC2CCCC2CNC(=O)CC=CC(C)(C)C)sc2ccccc12 c1(OC)ccc(C(=O)NC2CCN(C(C34C=CC(CC3)C4)=O)C2)c(F)c1 N1(C(C(NOC)=O)=O)CC2(CCCC2NC(=O)C2=CCCCC2)C1 N1(C(C2(C)CCC2)=O)CC=C(CNC(C2Cc3nnsc3S2)=O)CC1 CCCC(CNC(=O)CC1CCN1C(c1cccc(F)c1N)=O)CCC CC1(C)COCCC1C(=O)C(CC1CC(C(=O)NN)C1(C)C)=O.c1(C2CC2)cc(C)n[nH]1 C(=O)(CC(C)(C)CCC)NCC(CC=C)NC(c1cc2c(s1)CCSC2)=O C1(NC(C2(C)CC=CCC2)=O)CCN(C(c2cc(O)ccc2Cl)=O)CC1F CC1CCN(C(c2cccnc2N)=O)CC1CNC(C1(CO)COC1)=O N1(Cc2cc(C(=O)O)cc(Cl)c2)CCC2CN(C(c3ccno3)=O)CC2C1 C1(N(C)C(c2cc(C3CC3)ns2)=O)CN(C(C2(N(C)C)CCC2)=O)CC12CC2 C1(OCC)CCC(c2nc(-c3nc(C)cs3)nn2C2CCCC2)CC1 c1(C(=O)NC2C(CNC(c3ccc4snnc4c3)=O)C2)cc2c(Cl)ccnc2s1 c1(C(=O)NCC2(O)CN(C(c3cnc(CC)s3)=O)C2)ccc([N+](=O)[O-])o1 S(=O)(=O)(c1ccc(C(=O)NC2CCCC2NC(=O)COCC2CCCC2)o1)NC C(=O)(C(C)(O)C(F)(F)F)NCC1N(C(C2CCN(CC)C2)=O)CCCC1 c1(C(=O)NCC#CCNC(C(CC=C)C)=O)cc2c(=O)[nH]c(C)cn2n1 N1(C(CC(=O)NCC)=O)CCC2(NC(=O)Cc3cc(F)ccc3O)CC2C1 C1(NC(c2cccc(C(=O)NC)n2)=O)CCCN(C(=O)C(F)n2ccnc2)CC1 C12(CNC(Cn3cc(CCCC4N(C)CCC4)nn3)=O)CCC(CO)(CC1)CO2 N1(C(c2cnc(COC)s2)=O)CCC2(C1)CN(C(C1CCOC1C)=O)CCO2 C1(CC(=O)NC2(CCC)CCNC2=O)CN(C(c2c[nH]nc2CC)=O)CCC1C N1(C(C(C)CC2CCCCC2)=O)CCC(NC(c2cc(Cl)cc(Cl)c2)=O)C12CC2 C(=O)(CCCS(=O)(=O)N1CCCC1)N1C2CCC(NC(C3=CCCC3C)=O)(C2)C1 C1(NC(C(CCC)NC(C)=O)=O)CCCC12CN(C(c1cnn(CC)c1Cl)=O)C2 C1(CNC(CC)=O)CC(F)(F)CN1C(=O)C(C)C(F)(F)F Cc1ccnc(C(N2C(C(=O)NCCc3cccc(O)n3)CCC2C)=O)c1F n1(CCNC(C2(C)CCC2)=O)ccc(C(F)F)n1 N1(C(C2CC(=C)C2)=O)CC(C)(C)OCC1CNC(=O)COc1ccc(C)c(C)c1 C1(n2cc(C3N(C(CCCC=C)=O)CC3)nn2)COC2(CCC2)C1O CC1CCN(C(=O)NCCc2cc(C(F)(F)F)ccc2Br)C(C(=O)N(C)C)C1 CC(C)C(C)(CNC(c1cc(C2CCC2)no1)=O)NC(C1CC(F)(F)C1)=O C1(C(N2C(CNC(c3cc(C(F)F)cs3)=O)CC(O)C2)=O)CC2C=CC1C21CC1 c12cccc(c1)N(CCNC(c1cc(C)cs1)=O)C2=O.c1(N)ccc(C)cc1.CC=CCl C1(NC(C(CCC)C#N)=O)C2CCCN(C(=O)C3=CCSC3)C2C1(C)C c1(C(=O)NC(CCOC)C(=O)NCCN2CCC2)c(C)cncc1C C1(c2n(CC(=C)C)nnn2)(NCC2CCC3(CCC3)O2)CC2OC(C)(C)OC2C1 Cc1cccc(CC(=O)NC2CCC2NC(C23CC(F)(C2)C3)=O)c1Br C=CC1CN(C(c2cnc(OC)c(C(F)(F)F)c2)C(=O)NC2CCC2)CC1O N1(C(c2csc(O)n2)=O)CC2CCN(C(c3nc(Cl)cs3)=O)C2C1 C(CCC(C(=O)NC1CCCCCC1C)NC(=O)CC1CCOC1C)OC c1(OC(C(N2CCC(CNC(c3c(C)nc[nH]3)=O)C2)=O)(C)C)cccc(C#N)c1 c1(NC(C2(F)CCN(C(C=COCC)=O)C2)=O)c(C#N)cnn1C(C)(C)C Cc1ccc(COC(c2nn(C(C)(C)C)cc2Br)=O)c(F)c1 C1(NC(N2CC(NC(c3c(N(C)C)ccnc3)=O)C2)=O)C2Cc3ccccc3C12 Cc1nc(NC2CCCCC2NC(C2CCSC2)=O)c2c3c(sc2n1)CCC3 CC1CCN(N2CCCC2c2ccccc2)CC1C(N)=O c1(OC)cc(C(N2CCC(C)C2c2cn(CC(C)O)nn2)=O)ccc1C(C)(C)C C1(C(=O)NC2CN(C(c3c(OC)scc3)=O)CC2F)CC2(C1)CC(CO)C2 C#CC1(O)CCCN(C(=O)CNC(=O)CN(C(=O)CCC2CCCOC2)CC)C1 c1(C(N2CC(NC(C3(CCCC)CC3)=O)C(C)(C)C2)=O)cc2c(C)n[nH]c2cn1 C1(C(N2CCCC(NC(c3n(CC)c(O)nc3)=O)C2)=O)COC(C)(C)CO1 c1(CN(C(c2ccn(CCOC)n2)=O)C2CC2)cnc(-c2cncnc2)nc1 N(C(=NCCCn1cncn1)N1CCC(Oc2ccncc2)C1)CCF c1(C(=O)NC(CC)(C)CNC(=O)CCNC(N)=O)ccc(C(C)C)cc1C CCC(CC(=O)N1CCCCC(NC(c2cccc(C#N)n2)=O)C1)CC(F)(F)F c1(C(CNC(N2CCN(Cc3nc(C)[nH]n3)CC2)=O)=O)cn(C)c2ncccc12 C(C(C)(C)C#CC(=O)NCC1CCCNC1=O)NC(C(C(C)C)OCC)=O C1(COC(=O)Nc2c(C(=O)OCC)oc(Br)c2)CC(C)CC(C)(C)C1 N1(C(C2CC(C3CCC3)C2)=O)CCN(C(=O)CCC2CC2(F)F)C(C(C)(C)C)C1 C1(N(C(C(C)C)=O)CC(N2CC(C(O)C(=O)N(C)C)C2)=O)CCCCC1 C1(CNC(C2C(C)(C)C2CNC(=O)Cn2[nH]cnc2=N)=O)CCC(O)CC1 c1(C2C(C(N(CCC)CCNC(C3C=CCC3)=O)=O)C2)ccc(Cl)cc1 N1(C(CCN(C(CC2C(OC)CCCC2)=O)CCO)=O)CC2C=CCC(C2)C1 C(=O)(C1=C(Cl)CCOC1)NCC1C(C)CCN1C(C1(n2cccn2)CCCC1)=O S(=O)(=O)(c1scc(Br)c1Br)Nc1nn(C)c(C(F)(F)F)c1 c1(CNC(c2nc(C)oc2)=O)ccc(C(=O)NCCc2cn(C)nc2C)nc1 c1(C(N(CCC(=O)NC(CSC)C)C)=O)cc(O)cc(F)c1 c1(C(=O)NCC2(O)CCCN(C(c3c(OC)c[nH]n3)=O)C2)c(C)ccc(Cl)c1F C1(C(=O)NCC(C)(CO)NC(CC(CC)C)=O)CCN(OC)CC1 C(C(=O)NCCC1CCCN1C(c1cc(C)c(Br)o1)=O)(C(C)(C)C)OC C1(C)(C(=O)NCC(C)NC(C2(O)CC3CC2C3)=O)CC(C#N)C1 N1(C(c2cc(C)ncn2)=O)CCC2CN(C(c3cccc(C4CCC4)c3)=O)CC12 N1(C(CC2(C=C)CC2)=O)CCC(F)(CNC(=O)C(F)(F)c2cccnc2)C1 C(=O)(C1c2c[nH]nc2CN1C(=O)CC(CC)SC)N(CCOCC)CC C=CCN=c1[nH]cc(C(N2CC=CC2CNC(=O)C(CSC)c2ccccc2)=O)s1 N1(C(CN(C2CC2)CC)=O)CCC(NC(=O)Cc2csc(C)c2)C(CO)C1 c1(CC(C(=O)N2CC(O)(CCNC(=O)C3=CCC3)C2)OC)ccc(Br)cc1 O=C(NN1CCCC1C(N1CCC2CC1C(=O)O2)=O)c1nccs1 Cc1cc(C(=O)NC2CN(C(c3cnn(-c4ccccn4)c3)=O)C2)c(Cl)cc1F C1(CNC(Cc2cccc(CC)c2)=O)CN(C(=O)CC2CSC2)CCC1C C(CCC(=O)NC1CC1(C(=O)OC)COC)C.C1(OCC)CC1C(=O)NCC C#CCCC(C(=O)NCCCN1CCC1)NC(=O)CCOC(C)C CCC(C(C)(F)F)NC(c1conc1C(C)NC(=O)C(c1ccccc1)C)=O c1(C(=O)NC(CNC(CCCCC#C)=O)(C)CC)cc2cc(F)ccc2[nH]c1=O c1(OCCC(=O)NCC(=O)NC(CC=C)CC)ccc(Cl)c(F)c1 C(=O)(CS(=O)(=O)CCO)N(C1CCCCN(C(CC(n2ccc(C)n2)C)=O)C1)C C12(NC(=O)CCn3ccnn3)CCCC1N(C(=O)CCN1CCCCCC1)CC2 C12(C(=O)NC3(CC=C)CCN(C(C4C5CC(=O)CC45)=O)C3)CCN(CC1)CC2 N1(C(C2(C(CC)=O)CC2)=O)CC(CC(=O)N(CCC(O)CO)C)CC1(C)C c1(C(N(CCCNC(C23CC(C(C)C)(CO2)C3)=O)CC)=O)cc2ncccc2s1 Cc1c(C(=O)NCC2(C)CN(C(=O)CN3CCCC3)CCO2)ccc(F)c1F C1(NC(C2(N(C)C)CCCC2)=O)CC(NC(C23CCCC2C3)=O)C(O)C1 c1(-c2nc(C)c(Nc3ccc(Cl)c(C(=O)NCC4CC4)c3)s2)ccc2cn(C)nc2c1 CCC(F)(F)C(=O)NC1CC1CNC(=O)CCCOc1ccccc1Br C1(C(=O)NC2C(NC(COCC(=O)OC)=O)COCC2)Cc2nccnc2C1 Cc1cccc(C(O)C(=O)NC(C2CCN(C(C3(C4CC4)CC3)=O)CC2)C)c1F N1(C(C2C(CC)C2)=O)CC(NC(c2[nH]nnc2C)=O)CC1C N1(C(C(C)Nc2scc(C)n2)=O)CCC(C)(C)C(CNC(C23CC(C)C2C3)=O)C1 C1(NC(c2c(CC)occ2)=O)CCCCC12CCN(C(C1CCSCC1)=O)C2 CCCC(O)CC(=O)NC(C)(CNC(=O)C=CC=C(Cl)Cl)CO Cc1ncnc(C)c1CC(=O)NCC12CCCC1(C(=O)O)C2 c1ccc2c(c1)CC(=O)N2C.c1(C(C)C)cc(C(=O)NNC(=O)N(C)C)cc(Cl)c1 C(c1cc(Cl)sc1Cl)=CC(N1CCCC1c1ccc(F)nc1)=O C#CCCCCCC(=O)NCC1CC(C)CN(C(=O)CC2CCC(=O)CC2)C1 CCC(C)(CC)C(=O)NC(C1CCCN(C(=O)C(C)Sc2ccccn2)C1)C c1(N2CCC(NC(C3CC(C#C)(O)C3)=O)C(C)(C)C2)ncnn2c(Br)ccc12 C(=O)(CCC(CF)CF)NC(C(=O)NC(C)C(F)(F)F)C1CCOC1 N1(C(C(C(C)C)NC(CC(=O)NCC)=O)=O)CCC2(CCC2)CC1 C1(O)(C(=O)NC2CCC(CNC(C(C(=O)OC)C)=O)C2)CCCCCC1 c1(C(C2CC23CC3)N(CCCNS(C)(=O)=O)CC)ccccc1 c1(NCCN(C(=O)C(c2c(C)n[nH]c2C)C)CC)cc(C)ccc1[N+](=O)[O-] CCC(C)(CNC(=O)C(C)(C)CCNC(c1cn(C(C)C)cn1)=O)C(C)O C(=O)(C(F)(F)C1=CCOCC1)N1CCCN(CCNC(C(C)(C)C(N)=O)=O)CC1 S(=O)(=O)(CC(C#N)C1CCOCC1)N1CCCC(c2c(C(=O)OC)n[nH]c2)C1 N1(C(COCCOCC)=O)CC(NC(=O)C(c2ccc(F)c(Cl)c2)C)CC(F)C1 c1(C(N)=O)ccccc1C(=O)NCC1CN(Cc2ccncc2Cl)CCO1 C(=O)(C1=C(C2CC2C)N(C)C(=S)NC1c1c(C(=O)O)cnn1C)OCC c1(C(C(N2CC(O)(CN(C(C3CN(C(C)C)C3)=O)C)C2)=O)C)cccc(Br)c1 CCCC(C)CC(=O)NC(C)CC(C)NC(c1cc(Br)cnc1O)=O c1(SCC(N2CCC(CC)(NC(=O)C(Cl)=CCl)CC2)=O)nc(O)cc(C)c1C#N O=C(CC1=NNC(=O)C1)NCCC1CCCN(C(C2(C3CCOCC3)CC2)=O)C1 c1(CNC(C(=O)NCCC(=O)OC)=O)cncc(OCC(F)(F)F)c1 c1(C(=O)NCC(CNC(=O)CCOCC(F)(F)F)OC)cccc(Br)c1 C1(COC)(CNC(=O)CC2(O)CCCC2)CN(C(=O)CSc2nncn2C)C1 C1(NC(c2cc(C)c(=N)[nH]c2)=O)CC2CC(NC(C3CCSC3)=O)C1C2 c1(C(=O)NCC(C(=O)Nc2c(CC)n(CC)nc2)N(C)C)ncc(F)cc1F C1(C(N2CC(CC(C)NC(CNC(C)=O)=O)C2)=O)CC2(C1)NC(=O)NC2=O C1(NC(CCCCCC=C)=O)CCC2CCN(C(=O)CCC(C)(C)C)C1C2 C1(NC(C(C)C)=O)CC2CN(C(=O)C(c3cc(F)cc(F)c3)C)CC2C1 C1(CNC(c2n[nH]c(C)c2C)=O)CC2(CCC2)CN1C(=O)C=Cc1cscn1 C1(CC(=O)NCC2(CN(C(c3c(C)nco3)=O)C)CC2)CC(C)CC(C)(C)C1 C1(NC(COC(CC)(C)C)=O)CS(=O)(=O)CC1NC(=O)C(F)(F)c1cscn1 CC(C)(CCCNC(c1cc[nH]c(=N)c1)=O)NC(C1CCC12CCC2)=O c1(C(=O)NCC2CCN(C(Cn3nc(C)oc3=O)=O)C2)ncc([N+](=O)[O-])cc1C Cc1cc(S(=O)(=O)N2CCC(n3cc(C)nn3)CC2)c(C)cc1[N+](=O)[O-] C=C1CCN(C(=O)CNC(=O)C(C)(C)C)C(C(=O)NCC(C)CCO)C1 C1(C)(CNC(C2C(CC)C2)=O)CCN(C(=O)CC2CCCC2)C1 C1(C)(C(=O)NCC(C(C)C)(C)C)CC(O)CN1C(c1c[nH]c(=S)cn1)=O c1(OCCCOC)ccc(-c2ccc(NC(=O)C(C)CSC)cn2)cc1 c1(CC)onc(C(=O)N(CC(O)CN(C(=O)C(c2ccc(C)s2)C)C)C)c1C CC1(CNC(C2(C3CC3)CCC2)=O)COCCN(C(c2cccc(Cl)c2F)=O)C1 c1(NC(NC)=NCc2cnc(CC)o2)nc2ncccn2n1 N#Cc1c[nH]c(C(=O)NCC2CC(C(=O)N(CC3CC3)CC3CC3)CO2)c1 C1(F)(CNC(CCC2CC(OC)C2)=O)CCN(C(C2CCCC(C)(C)C2)=O)CC1 c1(-c2cn(C(C(=O)OCC)C)nn2)ccc2[nH]ccc2c1 C12(CNC(c3ccc(SCn4cccn4)o3)=O)COCCN1C(=O)COC2 C1(CCOC)(NC(=O)CC2NC(=O)NC2=O)CCN(C(C2(O)CCOC2)=O)CC1 C(C(C(=O)N(CCO)CC)NC(C1CCNC1=O)=O)OCC N1(C(C)=O)CCC2NC(=O)OCC2C1.C1CS(=O)(=O)N1CCC C(=O)(CC1=NN(C)C(=O)C1)NC(COCC)C(=O)NCC1(CCO)CCC1 C1(OC(=O)NC(C(=O)NCC)C2(C)CC2)CC2(CCCO2)C1 C1(C(=O)NCCN(C(=O)C(C2CCCCC2)C)CC)COCCC1(F)F C(=O)(C(CCF)NC(C1CC(=O)CCO1)=O)N1CCC(SC)C1 C1(NC(COCC(=C)C)=O)CN(C(C2(CN(C)C)CC2)=O)C2(CCCOC2)C1 C(C(=O)N1CC(CNC(=O)CCc2cncs2)CC1C)(C(F)(F)F)OC(C)=O C1(NC(c2cnc(C)o2)=O)CCC(CN(C(=O)C(F)n2ccnc2)C)CC1 Cc1cc(C(=O)NC2CC3CC2CN(C(=O)OC(C)(C)C)C3)c(F)cc1Cl c1(C(=O)NCC(C(C)C)NC(c2c(CCC)n(C)nn2)=O)cc([N+](=O)[O-])n[nH]1 Cc1nccc(C(=O)NCCN(C(=O)C(O)C(C)C)CC(C)O)c1N C(C)(CC(C)C(F)F)NC(C1(SC)CN(C(c2ccc(OC)nn2)=O)C1)=O C(=O)(CS(=O)(=O)N(C)C)N(CC(CC)NC(=O)C=CC1CCCC1)CC c1(OC)ccnc(C(N2CCC(NC(=O)C(C)(C)N(C)C)C2)=O)c1 Cc1cc2[nH]c(C(N3C4CCC3C(NC(C3C=CCC3)=O)C4)=O)cc2o1 c1(C(=O)NCC2=CCN(C(C(C)SC)=O)CC2)cccc2c1OC(C)C2 C(CCC(C)C(=O)NC1CCCC1NC(c1cnc(C)c(C(F)(F)F)c1)=O)OC N1(C(c2ccc(SC)s2)=O)Cc2ccnn2CC(NC(=O)COC2CCCC2)C1 C1(NC(C2(C)CCNC(=O)C2)=O)CN(C(C2(O)CC3CCC2C3)=O)CC2(CC2)C1 Cc1ccc2c(c1)SC(C(N1CC3(CCC(NC(c4cc[nH]n4)=O)CC3)C1)=O)C2 c1(CC)cc(F)ccc1C(=O)N(C1CCCN(C(=O)C(C)NS(C)(=O)=O)C1)C c1(C(N2CC(C=C)C(NC(c3ccn(CCC)n3)=O)C2)=O)cnn2c1OCCC2 c1(C(N2CC3C(C(=O)Nc4ncc(F)s4)(C3)C2)=O)cc([N+](=O)[O-])cs1 Cc1[nH]nc(Cl)c1C(N1CCCC1CNC(=O)Cc1csc(S)n1)=O CCCCCC(C)(CC)C(=O)NC1CCC(CN=c2[nH]cnc(Cl)c2CC)CC1 C1(CC=C)(NC(=O)CN(S(C)(=O)=O)C)CN(C(=O)C(F)(F)c2cccnc2)C1 C(=O)(C(C)CC(C)C)NC1C(CC(=O)N(CC=C)CCOC)CCCC1 C1(OC(C(=O)NCC)C)CCCCCC1.C12CCC1(C)n1cc(nn1)CNC2=O c1(C(=O)Nc2cc(OC(F)F)cc(N)c2)cccc2nc(O)ccc12 N1(C(c2nc(CC)oc2C)=O)CC2CC(C(=O)NCCOCCCO)C(C2)C1 Cn1c(C(=O)NCC2(O)CCN(C(C3(C4CCCO4)CC3)=O)C2)cnc1S N1(C(c2nc(CCC)sc2)=O)CCCN(C(=O)COCCOCC)C(C(C)C)C1 n1(CCN(C)C)ncc(C(N2CCC(Nc3ccccc3)CC2)=O)c1N C1(CC(=O)NCC(CC)NC(c2cc(C(N)=O)cs2)=O)CCC(C)CO1 C1(C(N)=O)CCCC(C(=O)NCCCCNC(=O)CCF)CC1 c1(C(=O)NCCC(C)NC(CCCCSC)=O)ccccc1S(=O)(=O)N(C)C C1(N(C(C(OC)OC)=O)C)CCC(NC(c2n[nH]cc2C2CC2)=O)CC1 N1(C(C2(CNC(C3(C)CCCOC3)=O)CC(=C)C2)=O)CC(C)CCCC1C N1(C(c2nc(C)oc2)=O)CCOCC1CNC(C1CC(=C2CC2)C1)=O C1(C(=O)Nc2nccs2)(Nc2[nH]nc(Br)c2-c2ccccc2)CCOCC1 CC1CCc2ncc(C(=O)NC(C)(C)CNC(C3CCC3n3cccn3)=O)n2C1 C1(CC(N2CCC(NC(C(CCSC)OC)=O)C2C)=O)CCCCC1(C)C N1(Cc2c(C)cccn2)C(=O)CCN(Cc2cccc([N+](=O)[O-])c2)C1=O CC1C(NC(=O)C=Cc2ccncn2)CCN1C(=O)CCOc1ccccc1Cl CCCCC(O)C(=O)N1CCC(C(C)(C)NC(C2(C(=O)OC)CCCC2)=O)C1 c1(CN(CCOC)CCNC(C23CCCC2C3)=O)cccc(OCC#N)c1 Cc1cc(C(=O)NC(CNC(c2snnc2C2CC2)=O)C2CC2)cc2ccoc12 CCC(C(=O)NCC1CCC(NC(=O)CCC=C(C)C)C1)C(F)(F)F c1(-c2cccc(OCCC)c2F)cccc2cc(C(=O)NCc3cc[nH]n3)[nH]c12 C1(CCO)CCC(N=c2[nH]c(NC3CC4C=CC3C4)nc3c2CCCCC3)CC1 N1(C(C(CCCC)CC)=O)C2CCC1C(CO)N(C(c1cc(OC)ncn1)=O)C2 N1(C(C(CCC)F)=O)CCC2CN(C(C3CCc4ncnn4C3)=O)C(C)C12 N1(C(C(C(=O)OC)C)=O)CCC(CCNC(C2CN(S(C)(=O)=O)C2)=O)C(F)(F)C1 c1(NC(C2(COC)CCCCC2)=O)ccc(-n2cncn2)c(F)c1 C1(C(=O)NC2CCC(C)(C)C2)(NC(Cn2ncc(C)c2)=O)CCCCC1 CC1OCCC1(F)C(=O)Nc1nc(Cc2cccs2)c(-c2nccn2C)s1 C(C(=O)NNC(=O)CCCOCCCS)SC(C)(C)C.C1CC1 c1(CC(=O)NC2C(NC(c3c(C)cn(C)n3)=O)CC2)ccc2n[nH]cc2c1 n1(C(C(=O)NC(C(=O)OC)C2CCCC2)C)cc(CCOC(=N)O)nn1 Cc1noc2nc(C(N3CCN(C(c4cccnc4S)=O)C(C)C3)=O)ccc12 C1(NC(C(C2CC2(Br)Br)N(CCCC)CCOC)=O)CCOCC1 C1(NC(c2c(OC)n[nH]c2)=O)CC2CCC1C(NC(=O)CC(C)C(F)(F)F)C2 Cc1nsc(N2CCC2CNC(=O)C2=CSCCO2)c1C#N c1(NC(=O)CCCC2CCCC2)cccc(NC(=O)C(C2CCCO2)C2CC2)c1 CC1(C)CN(C(C2CCCN2C=O)=O)CCC1NC(=O)CCN1C(=O)CCC1=O N1(C(C2N(C(C(COC(C)=O)C)=O)CCC2C)=O)CCCOCC1C c1(CC(=O)N(CC(C)O)CCNC(c2cnn(C(C)C)c2)=O)ccc(F)c(Cl)c1 C1(NC(C(c2cccs2)N(C=O)CCF)=O)CCN(c2ccccc2)C1 C(CCCCCC(=O)NCC1CCOCC1)NC(c1c(C)c(F)cnc1)=O c1(C(=O)NCCC2OCCN(C(CC(CC)C)=O)C2)c(O)cc(Cl)cc1F C=CCCC(C(=O)NCC1CCOCC1)N1CCOC(c2cn[nH]c2)C1 c1(C(N2C(CNC(C(C(C)C)(C)C)=O)C(C)(C)CC2)=O)ccnc2cc[nH]c12 C1(N(C)C)CN(C(c2cnn[nH]2)=O)CC1C(C1CC1)NC(=O)C(O)CC1CC1 C1(C2CCN(C(C3(C(N)=O)CC3)=O)C2)(NC(Cn2c(C(C)C)ncc2)=O)CC1 c1(OC)ccccc1C(C)C(=O)NC(c1cc[nH]n1)C1(C)CCC1 C1(NC(COc2cccc(C)c2)=O)CC2CC1CN(C(C1(C)CCC1)=O)C2 C1(CCCNC(c2n(CC=C)nnn2)c2cnn(CCOC)c2)CCC(C)(C)O1 CCCC(C)(O)CNC(C1CCC1NC(c1cc(CO)ccn1)=O)=O c1(C(=O)NC(C2N(C(CC3CC(=C)C3)=O)CCCC2)C)cccc2[nH]c(=N)oc12 c1(OC)cccc(C(C)=O)c1NC(C1CN(C(c2ncccc2C)=O)CCS1)=O c1(C(N2C(C)(C)C(NC(=O)CNC=O)CC2)=O)cnc(O)c2cccnc12 c1(NC(c2c(C)n[nH]c2)=O)ccc(Cl)cc1[N+](=O)[O-] CCC(C)CCCC(=O)NC1CC2(C1)CN(C(C1CCC1c1nncn1C)=O)C2 C1(CC(=O)NC(C(C)C)CNC(C2(C)CCOC2)=O)CC(=O)NC(=O)C1 C1(C(=O)NC(C)CCSC)(OC)CCN(C(c2nccnc2N)=O)C1 c1(OC)ccc(C(N2CCCC(NC(C3(C)CC(=O)N(C)C3)=O)C2)=O)nc1OC n1(CC)nnc2c1C(C(=O)N1CCc3cccnc31)CN(S(=O)(=O)CCCCl)C2 c1(C(=O)NCCC(C)NC(=O)Cc2cnccc2C(F)(F)F)snc(O)c1Cl C1(CC(=O)N(CCC(=O)NCC2CSCCO2)CC)CCCN(C)C1 c1(CCOCC(=O)N(C2CCN(CC3CCCCC3)C2)C)cccc(Br)c1 N1(C(c2c(COC)cccn2)=O)C2CCC1C(NC(=O)C=C(C)Cl)C2 C(C(=O)N(CCCCNC(=O)C(n1cc(Br)cn1)C)C1CC1)(C(C)C)SC N1(C(c2nc(CC)oc2)=O)CC2CCC(CNC(=O)CCc3cnccn3)C2C1 C(C(C)(CC)C(=O)NCC(C)(O)C(F)F)NC(C1C(=C)C1)=O N(C)(C1CCc2ccccc21)C(c1n[nH]cc1C)C(=O)NC(CC)(C)C N1(CC(CC)(C)N)CCCC(F)(c2ccccc2)C1 c1(C(N2CC3C(CNC(C(C)(C(C)C)NC(C)=O)=O)(C3)C2)=O)cnc2scnc2c1 N1(C(c2cnc(C(C)C)s2)=O)CC(C)CCC1CNC(c1ncc(N)cc1Cl)=O c1(OCC)ccc(C(=O)NC2CC2CNC(c2nnc(O)cc2C)=O)cc1Cl c1(COC)cc(C(=O)NCCC(=O)NC)n[nH]1.C12C=CC1C(=O)N2C1CC1 C12(CNC(C(CC)CN(C)C)=O)CN(C(c3cc(Cl)ccn3)=O)CC1CCO2 N1(C(c2c(CC)noc2)=O)CCC(C)(CC(=O)NC(C)CC2(O)CCC2)C1 C(=O)(C1=C(SC)CCCC1)N(C1CCN(C(C(CC)(C)OC)=O)C1)C CC1(C)CCC(F)(c2noc(CSC3CCCOCC3)n2)CC1 C1(NC(c2c(C)cc(C3CC3)cc2)=O)CN(C(=O)C(C)O)CC2(CC2)C1 N1(C(C2CCN(CC(C)C)C2)=O)CCC(C)(NC(c2ccc(OCC)o2)=O)CC1 c1(C(N(C2CCCC(NC(c3cnccc3Cl)=O)C2)C)=O)ccnc(S)c1 c1(C(N2CC(O)(CN(C(C(c3cnn(C)c3)OC)=O)C)C2)=O)cncc(Cl)c1C C(=O)(C1CCCn2nccc21)N1CCN(C(CNC(C)=O)=O)CC1 C=C(C)CC(C(=O)NC1CC(F)(CNC(=O)C(C)OCCN(C)C)C1)OC CCCC(CC)C(=O)NC1C=CCN(C(=O)CSc2ccc(OC)cc2)C1 C1(C(=O)Nc2ncc(C(C)(C)C)[nH]2)COC2(C)CC1C2 CCN=c1cc(-c2cn(C3CN(C(c4c(C)cccc4C)=O)C3)nn2)cc[nH]1 c1(C(=O)OC)cccc2c1CCC2NC(=O)C(C)(C(C)C)NC(C)=O c1(CC(=O)NC(CNC(CCc2ccc(C(=O)OC)[nH]2)=O)C)cnc(C)nc1O C1(NC(C(C)OCC#C)=O)CCCCN(C(=O)C(CC)CCOC)C1 C=C(C)C(C)(C)C(=O)NCc1nocc1C(=O)NCC1(CC2CC2)CCC1 c1(C(N2CC(C(C(=O)NCCCn3cncn3)O)C2)=O)cc2cccnn2c1 c1(SCC)ccc(CC(=O)NC2(C)CCN(C(=O)C(O)Cc3cnc[nH]3)C2)cc1 C1(NC(C2C(C)(C)CCN2C(C2CC=CC2)=O)=O)CCCOC12CCC2 c1(CC)n[nH]c(C)c1S(=O)(=O)NCC1CC(c2ccccc2C)C1 N1(C(C2(CC)CCCN2C(=O)CN=[N+]=[N-])=O)CC(C)CC(O)C1 CCCCCC(C)CC(=O)N1CCC(CCNC(c2c(C)ccc(Cl)c2N)=O)C1 C1(C(=O)OC)(CC)CCN(C(=O)C(C)N(C)C(C2(C)CC2)=O)C1 C(CN=c1nc(N2CCCC(CC3CC3)C2)c2c([nH]1)COC2)(C(F)(F)F)OC C1(C)(NC(CC2(N(C)C)CC2)=O)CCN(C(=O)C=CC2CCOCC2)CC1 c1(C(=O)NCC(C)NC(C2(C)CC2c2ccccc2)=O)coc2cccc(O)c12 N1(C(CSCC)=O)CC2CCCCC2(NC(c2cc(C3CCC3)nn2C)=O)C1 c1(OC)ccncc1C(=O)NCC1CC(F)CN1C(C1CCC(O)CC1)=O c1(C(=O)NC2(C(N3CCC(CC=C)C3)=O)CC2C)cc(O)cc(F)c1 C(=O)(CC(C)(C)COC)NC(CNC(c1[nH]cc(CC)c1)=O)C1CCC1 C1(=O)C(O)CCN1.C1(C(=O)N(CCC(=O)NO)C)CCN(CCF)CC1 c1(C(N(CC(C)SC)C)=O)cc(CO)n(C)n1.C1(=O)C=C(C)CN1 N1(Cc2cncc(NC(c3ccc(OC)c(I)c3)=O)c2)CCC(C)(C#N)CC1 C1(C2C(C(N(CCCN(C)C(C3CC3F)=O)C)=O)C2)CCCC1 c1(OC)cc(C(=O)N(CC(C)CNC(C2CCN(C)C2C)=O)C)cc(N)c1OC C12(C(N3CCC(NC(c4cccc(=S)n4O)=O)(CF)C3)=O)CCC(=O)N1CCS2 C1(C)(OCC)CN(C(=O)CNC(c2cncnc2)=O)C1.C12(CCC1)C(=O)N2 N1(C(C2CCCC(C(=O)OC)C2)=O)CCCC(C)(CNC(C2CCC(F)C2)=O)C1 C1(CNC(C(C)=C(CC)C)=O)CCC(NC(C2(N3CCCC3)CCC2)=O)C1 c1(NC(C2CC2c2c(F)cccc2F)=O)cc(Br)cc(Br)c1 c1(OCCCC)ccc(OC(=O)CN(C(C)CNC(=O)C(C)(C)C)C)cc1 N1(C(C2(c3cc(C)no3)CC2)=O)CCC2(CCC(NC(C3CCC(C)C3)=O)C2)C1 N1(C(C(CC)=CC)=O)CCC(C(C)(C)C)(CNC(=O)Cc2nncs2)C1 C(=O)(CCCCCSC)NCC(C1CCCCC1)NC(c1ccc(COC)[nH]1)=O C1(NC(c2c(CC)ccs2)=O)CN(C(=O)C=Cc2c(C)coc2C)CCC1F c1(C(=O)Nc2cc(O)c(Cl)cc2Cl)ccn2c(C3CC3)cnc2c1 C1(OC)CN(C(c2cccnn2)=O)C(C)(CNC(c2ccnnc2O)=O)C1 c1(C(=O)NC(C(C)NC(C2CCC(CC)O2)=O)CO)cccc(N(C)C)c1 Cc1ccc(C(=O)NC2CCCN(C(=O)C(C)(O)C3CC3)C2)c(C)n1 C(=O)(C(C)P(C)(C)=O)NCCCCC1CN(C(C2N(S(CCC)(=O)=O)CCC2)=O)C1 C(CC(C)C)(C(=O)NC(C)CS(C)=O)NC(CNC(CCC)=O)=O C1(C(=O)NC2CC(NC(c3cc(COC)no3)=O)CC2O)CS(=O)(=O)CC(=O)N1 C1(C(N2CC(CNC(C(C)OCC#C)=O)C2)=O)CC12CCOC2 C1(C(=O)NC2(C(=O)NCCC(F)(F)Cl)CSC2)CCCC12CCC2 c1(C(=O)NC(C2(C(N3CC4CCC3CC4)=O)CC2)C)cc(O)nc(O)n1 CCC(C)CC(=O)N1CC2CC2(NC(=O)C(C)(C)COC2CCCC2)C1 N1(C(C2=C(C)OCCS2)=O)CCC2CCCN(C(=O)C=Cc3ncc[nH]3)C2C1 Cc1cc(C#N)cnc1C(=O)NC(C)C(C)NC(=O)CS(=O)(=O)N(C)C Cn1cc(Cl)c(C(N2CCOC(CCNC(=O)CC3CCCC3O)C2)=O)n1 C1(CC(=O)N(CCOC)CCNC(=O)CC2CC2(Cl)Cl)CCC(=O)NC1=O C(CC(=O)NNc1nc(C(F)(F)F)cs1)c1nc(C#N)cc(C)n1 N1(C(CCCCC)=O)CC2(CCC2NC(c2ccc(Cl)c(F)c2)=O)C1 CCCCC(O)C(=O)NCC12CC(CC)(CN1C(=O)C(CC)N(C)C)C2 c1(C(=O)Nc2ccc(C3CCN(S(=O)(=O)C4CC4)CC3)cn2)cnn2ccccc12 N1(CCCC(=O)NCC2C(CNC(C3CC(C)(C)C3)=O)C2)C(=O)CNC1=O C1(CC(N2CCN(C(c3ccc(F)c(Cl)n3)=O)CC2)=O)CCC(F)(F)CO1 N1(C(c2ccc(N(CC=C)CC)cc2)=O)CCN(C(=O)CCC(N)=O)CC1C C1(C(=O)OC)(C(=O)NC2CCC(N(C)C(c3cnsn3)=O)CC2)CCOCC1 c1(C(N2CCC(N(CCC)C(c3c[nH]nc3C3CCC3)=O)C2)=O)nnccc1C c1(CC)ccnc(C(N2CCCC2CC(=O)Nc2cccc(OC)c2)=O)c1 N1(C(C(C2CN(C(C3C(C)CCOC3)=O)C2)O)=O)CCC(F)(F)CC1 c1(C(=O)NCCN(C(C(C)C2CCCC2)=O)C)cccc(C2CCC23CCC3)c1 N1(C(CCC(=O)OCC)=O)CCC(CNC(C2CC(O)C2)=O)C12CC2 N1(C(c2cccc(C)c2)=O)CCN(C(=O)C(C)(C)n2ccnn2)CC12CC2 c1(C(N2CCC(N(C(=O)C=C3CCOCC3)CCC)C2)=O)cc2sccc2n1C N1(C(C(CC)F)=O)C(CNC(=O)CNc2nccs2)CC2CC12 Cc1cc(C(N2CC(CNC(C3(c4ccc(Cl)c(F)c4)CC3)=O)C2)=O)ccc1Cl Cc1[nH]c2ccccc2c1CC(=O)NC(C)CCCNC(C12CC(C)(CO1)C2)=O CC1=CC(O)CN(C(C2(C)CCCN(C(=O)COCC3CC(F)(F)C3)C2)=O)C1 Cc1cc(C)n(CC(=O)NC2CC(CCNC(C3CCCCS3)=O)C2)n1 C(=O)(C#CC1CCOC1)NC1(C(N2CC(=C)C2)=O)CCC(C)(C)C1 c1(OC)c(C(=O)N(C2CCCN(C(=O)CCC3CC(C)(C)CO3)C2)C)csc1C CCC(C)C(C(=O)N1CC2C(C1)C2(F)F)N(C)C(C12CC1CNC2=O)=O N1(C(c2nccc(C)c2N)=O)C2CCC1CC(CNC(c1ccnc(F)c1)=O)C2 c1(C(=O)NC(CNC(c2cc(CO)[nH]n2)=O)C2CC2)c[nH]cc1-c1ccc(Cl)s1 C(=O)(C1CCCc2c1ncn2C)NC(CNC(Cn1c(C)ccn1)=O)(C)CO O=C(CC(CC1CC1)NC(C1CCC2(CC2)C1)=O)NC(c1ccco1)CO C#Cc1ccc(F)cc1C(=O)N(C1CC(NC(c2ccc(C)o2)=O)C1)C c1(C(=O)NCC(CO)NC(=O)CC2CC(=O)NC2=O)csc2nccn12 C(C(Cc1ccc(Cl)cc1)C(=O)N(CCCNC(=O)COCCF)C)OC c1(C(=O)NCC2CCC(C(=O)NCCCCCCO)CC2)cnc(O)nc1O C1(C(=O)NCc2cc(C)oc2)Cc2ccc(F)cc2C(=O)O1 c1(C(N2CCN(C3CN(C(C(C)(C)OCC)=O)C3)CC2)=O)nnc(O)cc1C c1(OC)ccc(F)cc1CCC(=O)NC1(CCNC(=O)CNC(C)=O)CCC1 C(CS(=O)(=O)C1CC1)NCC.C(CC=O)N(CC)CC c1(NC2C(C)CCN(C(=O)CCCC(N)=O)C2)cc(=O)n2cc(Cl)ccc2n1 c1(OCCCN(C2CC2(C)CN)C(c2cn(CCOC)nn2)=O)ccccc1Cl O=C1OCc2c(NC(C3(F)CCN(Cc4ccc(Cl)cn4)C3)=O)cccc21 c1(C(N2CCCC(C(C)(C)O)C2)=O)ccc(N=c2ccn3ncc(I)c3[nH]2)cn1 C=CCN=C(NCC(F)(F)C1CCC1)NCC(C)(F)F N1(C(C=C(C)C2CC2)=O)CCCC(C2CN(C(=O)C(F)=C3CCC3)C2)C1 S(=O)(=O)(CC(=O)NC1CCC(C(=O)N(C(C)C(=O)N(C)C)C)C1)NC C1(NC(CCN(CC)CC)=O)CN(C(=O)CSc2nncs2)CCC12CCC2 c1(C(=O)OC)cnc2c(Br)cncc2c1NCC1CC2CCCC(C1)C2 O=S(=O)(c1cc(Cl)cc(Cl)c1)N1CC2(CCN(c3nccc(Br)n3)CC2)C1 C1(F)(C(N(C2CCN(C)CC2)C)=O)CCCN(C(C2CC3(C2)CC32CC2)=O)C1 CCCCC(O)C(=O)NC(C)(C)CN(C)C(c1sccc1C(=O)OC)=O CC1=C(C(=O)NC2(C3CCN(c4cc(F)ncn4)C3)CC2)SCCO1 c1(C(=O)NC2C(C(=O)NC(C(=O)NC)C(C)(C)C)C2)cccc([N+](=O)[O-])c1Cl Cc1ccc2c(c1)SC(C(=O)NCC(C1CC1)NC(c1cc(C(F)F)no1)=O)C2 C=CC1(C(=O)NC2CCC(CCC(N3CCC(COC)C3)=O)C2)CCCCC1 C1(C(N2CCOCC(NC(C3(COC)CCCO3)=O)C2)=O)CCC2(CCC2)CO1 C1(C(=O)NC2CN(C(CCC(=O)N(C)C)=O)CC2O)CC(c2ccccn2)=NO1 CC(C)C(O)C(=O)NC(C)(C)C(C)NC(=O)CCCC1CCCC(=O)N1 n1(CCC)nnnc1C(c1csc(Cl)n1)NCC(C1CCCCC1)OC n1(CC(C)NC(C(C)NC(=O)NC)=O)cc(CN2CCCC2CO)nn1 C1(CNC(=O)CC(F)F)CN(C(=O)Cc2csc(-c3ccc(F)cc3)n2)CCO1 c1(C(=O)NCc2ncn(C)c2)ccc(-c2ccc3ncsc3c2)c2c1OCO2 C1(CNC(C(COC)n2cc(C3CC4(CCC4)C3)nn2)=O)C2CC3C1C3C2C(=O)O Cc1cc(C(=O)NC2CCCC(NC(c3[nH]nnc3C3CC3)=O)C2)c(N)c(F)c1 c12cn(nn1)CCSCCSC(=O)C2.CC(C)(C)OC(=O)CC(F)F c1(NC(C2N(C(CCOC)=O)C3C(C2)C3)=O)cc(F)c(Cl)cn1 CC1CN(C(c2sc(N(C)C)nc2Cl)C(=O)NCC2CCOC2)CCS1=O Cc1c(C(=O)NC2CCCC(NC(=O)C(c3ncccc3F)(F)F)C2)cnn1C CCC(C)CC(C)C(=O)NC(CNC(=O)Cc1ccc(F)nc1)C1CCC1 c1(CC)ccc(C(=O)NCCC(C)NC(=O)C(c2ccc(Cl)nc2)(C)C)nc1 C1(C(=O)NCC(=O)OCC)C2CCCC2CN1C(=O)CC1C=CCC1.C1CC1 S(=O)(=O)(c1cccnc1)C(N1CCC(CC(N2CC(F)(C(=O)OC)C2)=O)C1)=O C#Cc1ccc(C(N2CC(NC(=O)CC(=O)N(C)C)C3(CC3)C2)=O)nc1 CCCC(O)CC(=O)N1CC(CNC(c2cc(CC3CCC3)c[nH]2)=O)C(O)C1 C(=O)(C1=NN(C)C(=O)CC1)NCCOCCN(C)C(C1CCCC1(F)F)=O C(=O)(CCC(=O)c1ccc(O)cc1)NC1C(NC(Cc2cc(C)on2)=O)COC1 Cn1nc(C(=O)NC2(CCNC(=O)CC3CCNC(=O)C3)CC2)cc1CO C1(CCN(C)C(C23COC(CF)(C2)C3)=O)CCN(C(=O)CCC2CC2(Cl)Cl)CC1 C12(CNC(=O)CCOCCCNC(c3ccc(CO)o3)=O)CCC(CC1)O2 CN1CCCC(C)(C(=O)NCc2ocnc2C(N2CC(OCCO)C2)=O)C1 N1(C(Cn2c(C)cnc2)=O)CCOC(C(C)NC(c2ccn(CCC#N)n2)=O)C1 CC(C)(CS(C)(=O)=O)C(=O)N1CCN(CC(C)(C)NC(C2CCOCC2)=O)CC1 N1(C(c2cnc(COC)s2)=O)CC(C2CCCCN(C(C3(C)CC3(C)C)=O)C2)C1 CCC(O)C(C)C(=O)N1CC(C)(NC(c2cccc(C(N)=O)n2)=O)C1 N1(C(CCNC(CC(C)C)=O)=O)CCC(C)(NC(=O)CCC2CCCCC2)CC1 Cc1ccnc(O)c1C(=O)NC(C)CC1CCN(C(=O)C(C)C2CCC2)CC1 N1(C(Cc2c(C)noc2)=O)CC2(CCN(C(C3COCCO3)=O)CC2)CC1C C=C1CC2(C1)CN(C(=O)CN(C(=O)C(C)(C(C)C)OC)C1CCC1)C2 N1(C(C(CC)CO)=O)CCCCC12CC(NC(c1ccc3nc(C)cn3c1)=O)C2 C1(N(C(=O)CCn2ccccc2=O)C(c2ccc(Cl)s2)C)CC2CCC(C1)N2 N1(CCC)CCC(NC(C2CC(=O)CN2C(=O)CC2CC(N(C)C)C2)=O)CC1 c1(C(=O)NC2CCCN(C(C(C)CC3CCC3)=O)CC2)cccc([N+](=O)[O-])c1Cl Cc1cc(F)ccc1N1CCCC(NC(N2CCC(C(F)(F)F)C2C)=O)C1 C1(CC)CCCC1(C)C(=O)NCC1CC(F)CN1C(c1ccn(CCOC)n1)=O c1(C(=O)Nc2nc(C(=O)Nc3cc(C)cc(C)c3)n(C)c2)cc(C)c(C)cc1C c1(C(N2CCN(C(CCC)=O)C(Cc3ccccc3)C2)=O)c(Cl)ccc(F)c1N N1(C(c2ncc(NC)nc2)=O)CCCC2(CCN(C(C3CCCC(C)C3)=O)C2)C1 N(C(=NCCCF)NCc1cc(Cl)ccc1N(C)C)Cc1c(C)cccc1 N1(C(CCC2(N(C)C(=O)OC(C)(C)C)CCC2)=O)CCC(O)C(C)C1 C(=O)(C(F)(F)C(C)(C)O)NCCCCC(C)NC(C1C=CCCC1)=O c1(CC(=O)NC2(CC=C)CN(C(=O)C(F)(F)CNC)C2)c(C)nc2ccccn12 c1(OC)ccccc1S(=O)(=O)N1CC2C(C1)N2C(=O)Cc1cnc2ccccn12 N(C1CCCc2ccoc21)C(C1CC(O)(CNC(CN(C)C(N)=O)=O)C1)=O c1(NC(C2C3CN(C(C4CC(=O)NCC4)=O)C2C3)=O)cccc(Br)c1[N+](=O)[O-] C#CCCCCC(=O)N1CCCC(C)(NC(=O)CSCC(N2CCCCC2)=O)C1 c1(OC)ccc(C(CF)(OC)OC)cc1.C1(C(N(CCNC=O)CC)=O)CCCC1C CCCCC(CNC(C1C(Cl)(Cl)C12CC2)=O)NC(c1cnn(CC)c1)=O N1(C(CCN(CCCCC)C)=O)CCOCC12COCCN(C(=O)C=NOC)C2 c1(C(=O)NC2CCCC(NC(c3cn(C)nc3)=O)C2)cc(N)c(Cl)cn1 c1(C(=O)NC2CCN(C(c3[nH]c(=NCC)sc3)=O)C(C)C2)cc(C)c(Cl)cc1C N1(C(CCCOC)=O)CC2CCC(C1)N2C(=O)CCN1CCOCC1=O N1(C(CC2CC(CC)C2)=O)CC(NC(=O)CNC(=O)OC(C)(C)C)C(C(F)F)C1 c1(C(N(C2CCN(C(=O)C(C)SC)CC2)CCC)=O)cc(OC)cc(N)c1O N1(C(c2c(CC)nc(C)s2)=O)CCCC2C1CCN2C(c1cc(C)cc(C)n1)=O N1(CCn2c(C)c(Br)cn2)CCCC2C(NC(c3cc(Cl)no3)=O)C(C)(C)C12 C(=O)(CC(CC)CC(C)C)NC(CC=C)CNC(c1cc(C(C)(C)O)on1)=O CCCCC(O)C(=O)N1CC(CNC(c2sc(C(C)OC)nc2C)=O)C1 c1(C(N2CCC(N(C(=O)C(CC)CC=C)CC#C)CC2)=O)cc(C)c(C)cc1Cl Cc1[nH]nc2c1C(N(C)C(c1cn(CC3CCOC3)nn1)=O)CCC2 c1(C(C(=O)NCC(C)N(C(C2COCCO2)=O)CC)C)ccc(C(N)=O)cc1 Cc1ccc(C(=O)NC2CC(C)N(C(C3CC(=O)CO3)=O)C2)c2c1CCC2 C1(NC(C(CC)=CC)=O)CC2(CCC(NC(=O)CCS(=O)(=O)NC)CC2)C1 C1(OCC)CCN(C(=NCCc2ccccc2)NCc2cc(C)on2)C1 CCC(CC(=O)N1C2CCC(C2)C1CNC(c1ccncc1C(F)F)=O)C(C)C Cc1cccc(C(=O)NC(C(C)NC(C2(CO)CC2)=O)C(C)C)c1 N1(C(C=CCOC)=O)CC2CCC(C1)N2C(c1cc(C(C)(C)C)n[nH]1)=O C(C(C(=O)OC)NCc1ccc(CC)o1)SCC=C Cc1nn2ccccc2c1C(=O)NCC1CN(C(=O)C2=CC3C=CC(C2)C3)C1 CC1(C)CC(C(=O)NC2(C)CCN(C(C3CC4(CSC4)C3)=O)CC2)CC(C)(C)O1 N1(C(c2cc(F)c(I)c(F)c2)=O)CCC2(CCN(C(C3(F)CC3)=O)C2)C1 C1(NC(CN(C(=O)CCc2cc(OC)no2)CC#C)=O)CCC(C)C1 C1(C(=O)NCC2C(C)(C)C2)CN(C(=O)CC#N)C(C)(C)C1 c1(CC(=O)N(CCN(C(C(C)NC(=O)NC)=O)C)C)ccc(C(N)=O)nc1 c1(-c2ccc(C(=O)NC(CN(C(=O)COCCCF)CC)C)s2)cccc(F)c1 c1(C(C(=O)NC2C(CNC(C(c3cn(CC)nc3)=O)=O)C2)C)ccc(C)cc1 N1(C(c2n(C(C)C)ccn2)=O)CCCC(NC(c2ccc(Cl)cc2Cl)=O)C(F)C1 CCCC(C(=O)N1CCOC(CN(C(=O)C(F)CC2CCC2)C)C1)NC(N)=O C1(CC=CC)CCCN(C(=O)C(C)CN(C(=O)C(C)COCC)C)C1 Cn1ncc2c(O)nc(=NNC(=O)NCc3ccc(OC4CCCC4)c(F)c3)[nH]c12 c1(NC(C2CCCN(C(C(C)C(F)(F)F)=O)C2)=O)cnc2c(c1)CCC2 N1(C(=O)OC(C)(C)C)CCCOC(CNC(=O)CC2CC3(CC3)C2)C1 C1(NCc2nc(CCC(=O)NC)on2)CCC(N2CCCC2=O)CC1 CC1(C)CC(CNC(=O)CCc2cnco2)N(C(C2CCC2(C)C)=O)C1 C1(C(=O)OC)CCC(C(N2CC(CNC(=O)CNC(N)=O)C2)=O)C1 N1(C(C2CC(C(C)C)C2)=O)CC(O)CC1C(=O)NC1CCCCC1F C(=O)(C(C(=O)N1C(C(=O)O)CC1C)c1ccccc1)OCC Cn1cc2ccc(NC(=O)NCC3COCCC3c3ccccc3)cc2n1 N1(C(=O)CCc2cccc(O)n2)CC2(CCN(C(=O)C(F)CC3CCCC3)C2)C1 Cc1cc(Br)c2c(c1)CN(C(c1ccc(OCc3nn[nH]n3)c(F)c1)=O)CCO2 C1(CC=C)OCCC1(c1nnnn1C(C)(C)CC)NCCCC1CCC1 C1(C(=O)NCCOCC(N)=O)CC(NC(C2C=CCS2)=O)CCO1 C1(C(=O)NCCC(C)NC(=O)Cc2cncc(Br)c2)CCCC(=O)N1C CC(C)CC(C(=O)N1CCOCC1CO)NC(=O)CCC(N)=O c1(OCC=C)ccc(CC(N2CCC(NC(c3nc(=O)n(C)[nH]3)=O)C2)=O)cc1 c1(C(=O)NC2CCC(NC(C(C)NC(C)=O)=O)C2)cc(C)nn1-c1ccccc1 N1(C(C(CC)C(C)O)=O)CCC(C2(NC(=O)C=Cc3ccc(C(F)F)o3)CC2)C1 c1(OC)cc(N)c(F)cc1C(=O)NCC1(CF)CC2(CCC2)C1 C1(CC(=O)N(C)CC2CC(F)CN2)SC2=NCCN2C1=O.c1(C(=O)N)cn[nH]c1 C(C(=O)NOCC1CCCN1C)(c1ccccc1)NC(Cn1ccc(C)c1)=O C1(NC(c2c[nH]cc(C)c2=O)=O)C2CC3CN(C(c4cnc(C)n4C)=O)C1C3C2 C1(C(=O)NCC(CNC(c2c(CC)ocn2)=O)CO)CC(=O)N(C(C)(C)C)C1 N1(C(c2cc(CC)on2)=O)CCCC2(C(=O)O)CN(C(=O)CC(F)(F)F)CC2C1 C12(CNC(CCC(C)OC)=O)CCC(C1)N(C(c1cc(CN(C)C)c[nH]1)=O)C2 C1(C)(CNC(C=C(C)C(C)C)=O)CN(C(=O)Cn2cc(F)ccc2=O)C(C)(C)C1 n1(CC(=O)N(CCC(=O)NCC2CCC2C(=O)O)CCCO)cccnc1=O C1(CN(C(CNC(=O)OCC)=O)C)COCCN1C(=O)C(C#N)CC1CC1 Cc1cccc(C(N2CCC(NC(C3CC3c3cccc(F)c3)=O)C2)=O)c1 c1(N2CCC(Br)=C(C)C2)nc(=N)[nH]c(=NC(C)Cc2nncn2C)[nH]1 c1(C(=O)NCC23CC(NC(CSCCOC)=O)(C2)C(C)O3)c(Cl)ccc(F)c1N c1(CC(N2CCC(C(F)F)(CNC(c3coc(Cl)c3)=O)C2)=O)c(O)ncnc1O C1(NC(c2n(CC)ccc2)=O)CS(=O)(=O)CC1NC(c1cc(COC)cs1)=O C=C=CC(C)C(=O)NC(C)(C)CCNC(c1cc[nH]n1)=O Cc1nc(C(C)C)nc(O)c1C(=O)NC(C)C(C(C)C)NC(=O)C#CC1(C)CC1 C1(C(N(C(C)C(=O)O)CC(=O)NCCOC)=O)Cc2nccn2C1 N1(C(Cc2c(C)noc2)=O)CCC(NC(c2ccc(C(C)C)c(Cl)c2)=O)CC1C C1(NC(C2(NC(C=C(CC)CC)=O)CC2)=O)CC(C)(C)C12CCC2 O=S(=O)(c1cccc(=NCCN2CCCC2)[nH]1)NCC1CCC2CC12 C(c1ccc(C)cc1)=CC(N1CC(CCO)(NC(C(CC)n2ccnc2)=O)C1)=O N1(C(CC(CCC)O)=O)CCC2C(CCN2C(=O)CCCOCC2CC2)C1 C=C=CCC(=O)NCCCC(=O)NC(C)(C)COCC C(C(C)(C)C(=O)N1CC(CC(F)C(=O)NCC2(SC)CCCC2)C1)SC CCCCCCC(C)NC(c1coc(-c2cnn(C)c2)n1)=O C1(NC(CCC=C)=O)CS(=O)(=O)CC1NC(c1cnc(N(C)C)c(Cl)c1)=O Cc1cccc(C(=O)NC(C)CN(C)C(C2COC(=O)O2)=O)c1[N+](=O)[O-] C(CC(=O)N=c1ccn(C)[nH]1)N(C(=O)C(C1CCCCC1)=O)CC#C C(=O)(C1CCCc2nccn21)NC1(CNC(C2(SCC)CC2)=O)CCCCC1C c1(OC)cc(NC2CC(NC(C3(C)CC3Br)=O)C2)ccc1[N+](=O)[O-] C1(C)(C(=O)OC)CCN(C(=O)CCCSc2ccccc2OC(F)(F)F)C1 C(=O)(C(O)(C(F)(F)F)c1cn[nH]c1)N(CCCN(C(c1ccc(C)nn1)=O)C)C Cc1nc(C2CC2)ncc1C(=O)NC1CC2(C1)CC(NC(C1CCC1CF)=O)C2 c1(C(N(CCN(C(c2c(C)cc(CC)o2)=O)C)C)=O)nccc2ccccc12 c1(C(=O)NCC2(CN(C)C)CN(C(CC(C)C3CC3)=O)C2)cccc2c1CCC2 c1(C(N(CC(C)NC(C(CC)OC2CCCCC2)=O)C)=O)cc2c(ccn2C)[nH]1 CC1CCCN1CC(=O)NC1CC(CNC(c2nocc2-c2ccccc2)=O)C1 N1(c2nc(OC)cc(OC)n2)CC2(CCOCC2)CC1C(=O)NC1CN(C)C1 Cc1nnc(NCC2CCC(CNC(c3c[nH]ccc3=O)=O)CC2)c(C#N)c1C c1(CNC(CCCSC(C)C)=O)ccccc1-c1cn(C2CCCC2)nn1 C1(NC(CC2C(NC(c3cc(CCC)[nH]n3)=O)CCCC2)=O)CCC(C2CC2)C1 CCC1=NOC(CC(=O)NCC=CCC(=O)NCCOCC(F)F)C1 C(=O)(CC1=CCCC1)N(CC(C)NC(=O)C(c1ccc(O)cc1)C)CC CC1Cc2cc(C(=O)NCC3COCCN(C(=O)CCS(C)(=O)=O)C3)ccc2O1 C(c1ccc(F)cc1)=C(C)C(=O)N(CCC(O)C(C)(C)C)Cc1nn[nH]n1 Cc1coc(C2CCCN2C(c2cscc2Br)C(=O)NCCCOCC2CC2)n1 C1(CNC(=NCC)NC2CCN(C(=O)C3CC3)CC2)C(F)(F)C12CCCC2 N1(C(C2CC(C#N)C2)=O)CC2CC(NC(c3cc(F)cc(F)c3)=O)C1C2 c1(OCOC)ccc(C(=O)NC2CC(F)(CNC(c3cnc(S)[nH]3)=O)C2)cc1 C(CC(=O)NC1CC(NC(C23CCC2C3)=O)C1)N(CC)CC CC1CC(C(=O)NC(C)CCNC(=O)C=CC2CCCC2)CCS1(=O)=O N1(C(C(C)(C)c2ccns2)=O)C2CCC1CN(C(C1CC1CN(C)C)=O)C2 c1(OC)ccc2cc(O)c(-c3c[nH]nc3C(N3CCCCNC(=O)C3)=O)cc2c1 CC(C)C(C(=O)NCCCCNC(c1cnc(Cl)[nH]1)=O)c1cnn(C)c1 C1(CCN(C(C(C)OC)=O)C)CCN(C(c2ccc(C(F)(F)F)cn2)=O)CC1 Cc1cc(C(N2CCC3(NC(c4ccsc4Cl)=O)CC3C2)=O)c(C)n1C Cc1cnn(C(C)C(=O)NCCN(C)C(C2CCN(c3nncs3)C2)=O)c1 C(C(C(=O)NCCC1CCN(C(=O)C=CCn2cncn2)C1)OC)OC c1(CN(C(N(CC(O)CO)CC)=O)Cc2ccc(F)cc2)nc(Cl)oc1C C#Cc1ccc(F)c(C(=O)NC2(C3CC3)CCN(C(=O)C(O)CCCC)C2)c1 N1(C(c2cc(C)sc2C)=O)CCC(NC(=O)C2=CSCS2)C(F)C1 C(=O)(C(=O)CC(C)CC)N1CC(NC(CC2CC(=C)C2)=O)C(SC)C1 C12(C(=O)NC(c3ncc[nH]3)CC)CC(CN1C(=O)CC(C)OC)C2 C1(C(=O)NCC2(C(C)(F)F)CC2)CCCN1C(C1CC1C1CCCC1)=O CC1C2CCC(C2)C1C(=O)N(CCCC(=O)NCCOCCO)C C1(C(N2C(C)CC2)=O)CCC(NC(=O)C(C)Cc2ccccc2)CC1 C1(C(N(C)CCNC(c2coc(Cl)n2)=O)=O)OCCOC1(C)C c1(C(N2CCCC(CN(C(C(CC)C#N)=O)C)C2)=O)c(C)ncnc1C C(C)(C(=O)N1CCC(O)(CN(C)C(c2cc(C)co2)=O)CC1)(C(C)C)NC(C)=O CC(C)CC(C)CC(=O)NCC1(O)CCN(C(=O)C(F)(F)CO)C1 C(=O)(C1=CCOCC1)N(C)CC1CCN(C(c2nn(CC)c(C3CC3)c2)=O)C1 N1(C(c2c(C)ccc(C)n2)=O)CC2(CC(C(=O)NC(CO)CC(C)(C)C)CO2)C1 C1(OC(C)C(=O)N(CC(O)CNC(c2ccc(=N)[nH]n2)=O)C)CCCCCC1 Cc1cccc(CCC(N2CCCC2CNC(C2CC3CCC2O3)=O)=O)c1 c1(CC(N2CCC(C(C(=O)NCc3cnccc3Cl)F)C2)=O)ccc(Cl)cc1 N1(C(C2N(C=O)CCC2)=O)CCC2(CC1)CC2NC(c1cccc2ccoc12)=O c1(CN2CCN(C(=O)C(Cl)(Cl)Cl)C(C(F)(F)F)C2)c[nH]c2c([N+](=O)[O-])cccc12 CC(C(=O)NCCC1(NC(C2CC=CC2)=O)CC1)N1CCCC1 N1(C(C2(C)COC2)=O)CCC2CCCN(C(=O)CS(C)(=O)=O)C2C1 C(c1ccccc1C)=CC(=O)N(C1CCN(C(C(C2CC2)OCC)=O)C1)CC c1(NC(C(=O)N(CCC)CCNC(=O)NCC(F)F)=O)ccc(C)cc1Br c1(OCC)ccc(SCC(N2CC3C(N(C(=O)C(C)C(F)F)C)C3C2)=O)nc1 c1(CCCC(=O)NCC2N(C(C(CC)NC(N)=O)=O)CCC2)ccc(Br)cc1 N1(C(C2(OC)CCSC2)=O)CC2(CC(NC(=O)Cn3nnnc3C3CC3)CO2)C1 C(N=c1cc(NCCCCN(C)C)nc[nH]1)C1(OC(C)C)CCSC1 CCCCCCCCNC(=O)C(C1(O)CN(C(c2n[nH]c(=N)[nH]2)=O)C1)F C(=O)(CCC(C)C)NCC(N1C(CN(C(C(C)(C)SC)=O)CC2CC2)CCC1)=O CC1(C)CCC(CN=c2nnn(-c3ccccc3)[nH]2)(NCc2ccco2)CC1 N1(C(CCS(=O)(=O)N(C)C)=O)CCC2(CC(NC(C3C=CCCC3)=O)C2)C1 N1(C(C(C)(C)c2cncnc2)=O)CC2CCCC(C1)N2C(=O)CN1CCCCC1 C(=O)(CC(O)CCCCC)NC(C1(O)CN(C(CCC(=C)Br)=O)C1)C C1(CNC(C2CCCO2)=O)CCN(CC2C3CNCC23)CC1 Cc1cc(Cl)c(C(=O)NC2CCN(C(=O)Cc3ccc(C)o3)CC2O)cn1 c1(C(N2CCN(C(c3cn(C(C)C)nn3)=O)C(C)C2)=O)cc2cccc(Cl)c2s1 C1(C#N)(C(N2CCC(O)(CNc3ncc(C)cn3)CC2)=O)C(C#N)C1(C)C C12(C(=O)OC)CCC(C(=O)NCC3(C)CCOC3)(CC1)CC2.C(CO)O c1(C(N(CCC)CCNC(C2(CCOCC)CCCC2)=O)=O)nc(Cl)c(CC)[nH]1 C1(F)(C(N2CC(OC)C(NC(=O)C(C)c3cccs3)C2)=O)CCN(C)CC1 c1(-c2cn(CCc3cc(C)no3)nn2)ccc(CNC(=O)CC2CCCO2)cc1 N(C1Cc2ccccc21)C(C(=O)Nc1cncc(C#C)c1)=O C1(C(N(CC(C)(C)NC(C2CC(=O)NC(=O)N2)=O)C)=O)CCc2cnnn2C1 N(C1CCCc2c1cnn2Cc1ccccc1)Cc1ccc(CN)cc1 C(=O)(CC(C)(C)C1CCCCC1)N(C1CCN(C(=O)C=Cc2ccncc2)C1)CC c1(C(N2CCC3CN(C(C4C(CN(C)C)C4)=O)CC32)=O)cc([N+](=O)[O-])cnc1O C(C(=O)NC(C(=O)NCCCn1cncn1)C1CCC1)(C(C)C)SCC N1(C(C2(C(=O)NC)CC2)=O)CCC2(CC1)CC2C(=O)NCCC1CCCCCC1 c1(NC(C(c2cc([N+](=O)[O-])sn2)N(c2nncs2)CC)=O)ccc(OC)cc1C C1(C2CCN(C(=O)CCP(C)(C)=O)C2)(NC(CCOCC)=O)CC1 N1(C(C(C)(C)CO)=O)CCC(O)(CCNC(C2(C(N3CCCC3)=O)CC2)=O)CC1 CCCC(C)(C)C(=O)N1CCC(O)(CNC(=O)Cn2c(C)c(C)sc2=O)C1 N1(C(Cc2nc(C)sc2)=O)CCCC(C)(C)C1CNC(C1(C)CCNC1=O)=O Cc1nc(C)c(C(=O)NC2CCC(NC(C3CC34CCCC4)=O)CC2)s1 c1(C(=O)NC2CCC(N(C(c3c(C)cccn3)=O)C)C2)cc(N)cc(O)c1C C1(CC(c2noc(CN(C)CC)n2)C)CCCN(C(=O)CC2CC3(N)CC2C3)C1 N1(C(c2scc(C)c2)=O)CC2(CCNC(c3ccc(Cl)cc3)=O)CCC1C2 Cc1nocc1CCC(=O)NC1(CCNC(=O)CCC2CCCCO2)CCCC1 C(CC(C(=O)NCc1ccc(Cl)cn1)NC(=O)CCOC(C)C)=CC CCCCC(CN=c1[nH]c(C)nc(C)c1F)NC(c1ccncn1)=O Cc1ccc(C(N2CC(C(N3CC4CC4C3)=O)C(F)(F)C2)=O)cc1C#N N1(C(C(Cn2ccc(C)n2)C)=O)C2CCC1C(C)C(NC(=O)CC1CC=CC1)C2 c1(C(=O)OCC)ncc(CNC(C)C(C)O)cn1 Cc1cc(Br)sc1C(=O)NCC(C)NC(=O)CCc1ccco1 CCCC(CCC)C(=O)NCc1nc(C(N2CC(COC)C2(C)C)=O)co1 N1(C(c2c(C)cccn2)=O)C2CC=C(C(=O)N3CC(O)(c4nn[nH]n4)C3)C1CC2 c1(N2CCC(=C)C2)cc(N2CCC(C(N)=O)C2)ncn1 NS(=O)(=O)c1coc(C(=O)NC2CC(NC(C3CC4(CC4)CO3)=O)C2)c1 c1(CC(=O)N(CC)CC2CCN(C(=O)CC(C)OC)CC2)cccc(F)c1Cl c1(C(=O)NCC2C(NC(C(N3CCOCC3)C)=O)CCC2)cocc1C(N)=O c1(C(N(C)Cc2c(C)ncs2)=O)c(-c2ccccc2)nn(C)c1Cl c1(OC)cccc(Cl)c1C(N1CCC(NC(c2nc(C)ncc2Br)=O)C1)=O C12(OC)CCCC(CC(NC(=O)Nc3ccc(SC)nc3)C1)C2 N1(C(COC(CC)(C)C)=O)CCC(NC(c2c(Br)nnn2C)=O)CC1 N1(C(c2c(NC)cnnc2)=O)CC(C)CN(C(c2cncnc2C)=O)CC1C C=CCCC(C)N=c1nc(N2CCn3cnnc3C2)c2c([nH]1)CCC(C)C2 C1(CNC(CCN(CCC)C)=O)CC2CCC(C1)N2C(=O)C(C(C)OC)N(C)C C1(NC(c2cn(CC=C)nn2)=O)C2CC1N(C(=O)CN(c1ccc(Cl)cn1)C)C2 c1(C(C(=O)NC2CCC2)N(C(CCSC)C)C)cc(S(C)(=O)=O)c(C)o1 c1(-n2ccc(C)c2)ccc(C(N2CC(NC(c3cc(C)co3)=O)CC2C)=O)cc1 c1(C(=O)NC2CN(C(c3nc4ccccc4o3)=O)C2)ccc2c(c1)CCNC2 N1(C(c2cn(CC=C)nc2)=O)CCN(C(c2csc(Cl)n2)=O)CC(O)C1 C=C1CCC(C(N2CC=CC(NC(=O)C(C)CSc3ccccc3)C2)=O)CC1 C1(NC(C(COC)COC)=O)CCCCN(C(=O)C=Cc2ccccc2)C1 c1(C(=O)NC2C=CCN(C(C3CCC(C)(C)CC3)=O)C2)ccc2cnoc2c1 C1(C(N(C(C)C)C)=O)CCN(C(=O)C(N2CCN(c3nccnn3)CC2)=O)CC1 C1(C(=O)NCC2OCCN(C(c3ccc(=N)[nH]c3)=O)C2)Cc2ccc(F)cc2O1 Cc1cc[nH]c1C(=O)NCCCCCNC(=O)C(=O)NCCc1ccccc1 N1(C(Cn2c(C)nnn2)=O)CCC(C2CCCN2C(C23CC(CO2)C3)=O)CC1 CCC(CC(=O)N1CCCC(NC(=O)Cc2ccn(C(C)C)n2)CC1)C(C)C C1(C(=O)NC2CC(NC(C(C)NC(=O)C3CC3)=O)CC2O)CCCC12CCC2 c1(C(N2CC3C(CNC(C4CCC(C(N)=O)C4)=O)(C3)C2)=O)cc(O)ccc1F Cc1nc(C(C)C)sc1C(N1CCC(CNC(c2c[nH]nc2F)=O)C1)=O n1(CC)nc(C)c(CC(N2CCOCC(NC(=O)CC(C)O)C2)=O)c1C N1(c2ncc(C#C)cn2)CC2(CN(C(c3cccnn3)=O)CC(C)(C)O2)C1 CC(CF)C(=O)NC(C)CCNC(=O)CCNC(c1ccco1)=O c1(C(=O)NC2C(C)CN(C(=O)Cc3ccn(C)n3)C2)ccc(O)c(C(=O)O)c1 C1(C(=O)OCc2n(-c3cn(C)nc3)cnc2)CCCCC(P(C)(C)=O)C1 C=CCC(C)(CC)C(=O)NCC1(C)CC(C(=O)NC2(c3ncccc3Cl)CC2)C1 C(=O)(C(CCC)NCC(C1CC1)OC(C)=O)NCC=C CCCCC(CC(=O)NCCC1CC=CCC1)NC(c1cccc2ccoc12)=O N1(C(C2CC(O)(CNC(C3(COC)COC3)=O)C2)=O)CC2CC2C2CC12 N1(C(CC)C(=O)NCCOC2CN(C(c3ccon3)=O)C2)C(=O)CCC1=O CCC(C)C(C(=O)N1CCCC(CCNC(=O)CCCCSC)C1)OC N1(C2CC(CC(=O)OC)C2)C(=O)C2CCCCN2C1=O Cc1onc(-c2ccc(F)cc2)c1C(=O)NCC1(CO)CCCNC1 c1(C(N2CCC(CN(C)C(C3(F)CC4(CCC4)C3)=O)C2)=O)cncc2sccc12 C1(NC(c2cnc(SC)s2)=O)CCC(C)(CNC(=O)CCc2cccn2C)C1 N1(C(C2N(C)CCC2)=O)CCCOC(CNC(c2cc(C(C)(C)C)n[nH]2)=O)C1 Cc1ccc(C(N2CC3C(CNC(C4(C)CCC(=O)NC4)=O)C3C2)=O)c(F)c1C c1(NC(C2(F)CCN(C(Cc3nc(C(C)=O)on3)=O)C2)=O)cc(C)cc(Br)c1F N1(C(c2c(CC)occ2)=O)CCN(C(=O)C(C(C)(C)C)NC(N)=O)C(C)C1 C(CN=c1c(Br)c[nH]cc1[N+](=O)[O-])=C1CCC(NC(C=COCC)=O)C1 C1(C(=O)NC(C(=O)NCCC(C)(O)C2CC2)C2(O)CCC2)C2C3CCC(C3)C12 C1(C(=O)NCC(CC(C)C)C)C2CC(O)C(C2)N1C(=O)C(C)CC1CCC1 C1(NC(c2ncc[nH]c2=O)=O)CN(C(=O)C2=CCOCC2)CC(F)(F)C1 c1(NC(C)=O)cccc(NC(=O)C(C)(C)CNC(=O)CCCC2CCCO2)c1 C(CC(F)F)(C(=O)NC1CC(C)(C)C12CC2)N(C(Cc1c(C)n[nH]c1)=O)C Cc1ccc(C(=O)NCCC2CCC(NC(=O)C(=O)NCC(F)(F)F)C2)s1 c1(C(N2CCC(CCNC(C34CC(O)C3C4)=O)C2)=O)cc(-c2ccco2)[nH]n1 N1(C(C(C)Oc2ccccc2)=O)CCN(C(C2CC3(CC(=O)N3)C2)=O)C(C)C1 CC1(C)CCCCC(C(=O)NCCNC(C23COCC2C3)=O)C1 CCC(C)C(O)CC(=O)NC(Cc1cn[nH]c1)C(=O)NCC(C)N(C)C C1(NC(C(C)O)=O)CC1C1CCCN(C(c2cn(C)nc2C2CCC2)=O)C1 N1(CC=CC(=O)N(CC(CC)NC(=O)Cc2csc(S)n2)C)CCOCC1 c1(C(=O)NCC2(CNC(C34CC(C)(C3)C4)=O)CCCC2)cc2n(n1)CCNC2=O c1(CNC(CNC(=O)NC)=O)cc(C(=O)NC(C2CCOC2)CC)n[nH]1 c1(C(=O)NCCCCNC(c2cnc(C)s2)=O)cccc(-n2cncn2)c1 N1(C(C=CCOC)=O)C2CCC1C(F)C(NC(C1CC=CCC1)=O)C2 CC1(CC(=O)NCC#CC(=O)NCC(O)CNC(N)=O)OCCO1 C(CC(O)C(=O)N1CC2CC2(C(=O)NCCCc2ccccn2)C1)SC CC(C)(F)C(C)(F)C(=O)NCC1CC(NC(=O)CCc2ccc(Cl)nc2)C(O)C1 Cc1cc(C(=O)N(CCCCN(C(=O)C(C)C(F)F)C)C)oc1C c1(N(CCC#N)C)ccc(S(=O)(=O)NC(c2cccnc2)(C)C)cc1F C1(OC)CCN(CC(=O)NC(CNC(=O)CN2CCC(C)C2)C(C)C)C1 CC(O)C(C(N)=O)NC(C1CCC(NC(=O)CCc2cccnc2)CC1)=O N1(C(CC(C(=O)OC)C)=O)CC(CNC(=O)Cc2ccccc2Cl)C2(CCC2)C1 N1(C(C(c2cnn(C)c2)NC(COCCCCC)=O)=O)CCC(CO)CC1 CCC(CC)C(C)C(=O)N1CC2CCCC2(NC(c2cnc(Cl)[nH]2)=O)C1 c1(CNC(N2CCCC2)=O)ncccc1S(C)(=O)=O.CCCCCN c1(CC)cccnc1C(N1CCCC1(C)CNC(=O)C(C)(C)c1ccccn1)=O C(=O)(C1=NOC(C)C1C)N1CCC(CC=C)(C(N2CC=CC2)=O)C1 C1(CCOC)(NC(=O)C=C(C)Cl)CCN(C(=O)CCC2C(=O)NN=C2C)C1 C(=O)(CC(O)C(C)C)N(C)CC1CCN(C(C2(CCOCC)CCC2)=O)CC1 C1(CNC(C(C(C)C)O)=O)CCC2(CO1)CC(NC(=O)Cc1cc[nH]n1)C2 c1(C(=O)NCCC2CCN(C(C3N=C(C)SC3)=O)CC2)c(Cl)ccc2ccoc12 c1(C(N2C(CC)COCC2)C(=O)NC(c2ccccc2)C)cccc2c1CCC2 C(=O)(CS(=O)CCC(F)(F)F)NCC1CCN(C(Cc2cn(C)nc2)=O)C1(C)C c1(CSCC(=O)NCCC(C)NC(CCC#CC)=O)ccc(Cl)cc1Cl N1(C(=O)OC(C)(C)C)CC2CCC(CNC(=O)NCCN3CCC(C)(C)C3)C2C1 C(=O)(C(CCC)CC(C)C)NCC1(OC)CN(C(c2cn(CCCC)nn2)=O)C1 c1(OCC)ccccc1CN(CCCNC(=O)C(O)CC1CCCCC1)C(C)C C1(CC(=O)NC2CC(OC)C2)CN(C(=O)CN=[N+]=[N-])C(C)(C)C1 N1(C(c2ccc[n+]([O-])c2)=O)CCC2(CCNC2=O)C1 c1(C(=O)NC2CCCN(C(=O)C(O)CC(F)F)C2)cc2c(nc1O)CCCC2=O N1(c2ncn(C)c(=O)c2)C2CCC1CN(C(c1ccc3c(ccn3C)c1)=O)CC2 CC(C)C(C)C(CNC(c1nocc1Cl)=O)NC(=O)CSCc1cccs1 C(=O)(C1CCc2cc(F)ccc21)NCC(CO)NC(c1c(C)n2c(n1)scc2)=O N1(C(C23CCC(OC)C2C3)=O)CC(C)C(C)(C(=O)NCC2CC(=O)N(C)C2)C1 Cc1noc(CNC(c2ncsc2Br)c2nnnn2CC2CCCO2)n1 C(c1ccccc1OC(F)(F)F)=CC(=O)NC1C(NC(C2CC(C)(F)C2)=O)C1 c1(N2C(CNC(c3cc(Br)ccc3Br)=O)CCCC2)ccn2ncc(Br)c2n1 c1(C(N2CCC3(CN(C(C4(F)C5CCCCC45)=O)C3)C2)=O)cc2scc(Cl)c2[nH]1 CC1CC(NC(=O)C2=CCC2)CN(C(c2ccc(Cl)c(N)c2)=O)C1 Cn1nccc1C1CC1C(N1CCC(CNC(=O)CSCC(=O)OC(C)(C)C)C1)=O N1(CC(=O)NC(CC)CNC(=O)CC2(O)CCCC2)CCCCC1CO N1(C(C2N(CC)CC2)=O)CCCCC1CNC(c1ccc(OC(F)F)cc1)=O C1(NC(CC2(C)CC2(Cl)Cl)=O)CCN(C(C2Cc3cscc3C2)=O)CC1F C=CC1CC(N=c2ccc(Br)c(S(=O)(=O)N3CC45CCC4(COC5)C3)[nH]2)C1 C1(N(C(CC(c2cccc(F)c2)C)=O)C)CCC(NC(=O)COCC(F)F)CC1 CN1CCCC(O)(CC(=O)NCCN(C)C(C2(CCO)CC2)=O)C1 C(=O)(C(C)CS(C)(=O)=O)NCC(c1cccc(C)c1)NC(C1(O)CCCC1)=O CN1C(=O)CCC1C(=O)NC(C(=O)NCCCOCCO)C1CC1 c1(NC(c2cncc(-c3cc4ccccc4[nH]3)n2)=O)cc(F)ccc1[N+](=O)[O-] CCC(CC(=O)NC(C(=O)N1CC(C(N)=O)(OC)C1)C(C)C)SC CC1(C(N2CC(NC(c3cccn4nncc34)=O)C2)=O)COc2ccccc2O1 N1(C(C(N2CC(CCNC(=O)C(C)CO)(OC)C2)=O)C)CCc2ccccc21 S(=O)(=O)(c1ccc(N2CCCOC(C)(C)C2)c(F)c1)NC(c1nncn1C)C C1(NC(c2cccc(CNC(C(C(C)C)(C)O)=O)n2)=O)CC2CCC(C1)C2O c1(C(N2CCCC(CC)(NC(=O)C3=NNC(=O)C3)C2)=O)cccc(S(C)=O)c1 C(CCCCCCCCCO)n1cc(-c2c(F)ccc(I)c2)nn1 S(=O)(=O)(c1cccc(C(=O)NCCNC2CCCCC2)c1)NC1CC(=O)C1 Cn1cc2cc(C(N3C4CN(Cc5c(O)cccc5O)CC34)=O)ccc2n1 N1(C(c2c(OCCOC)nccc2)=O)CC2CN(C(C3CC(O)C3)=O)C2C1 C1(NC(C2(CC)CC2)=O)(Cc2ccccc2)CCCN(C(=O)CC(C)C(F)F)C1 C1(CC(=O)NCC(CCC)NC(c2csc(C)c2OC)=O)CCS(=O)(=O)C1 c1(C(=O)NCC2C(NC(c3cc(CC)on3)=O)COC2)ncccc1S(C)(=O)=O C(=O)(CC(C)CC(C)C)N1C(C)(CCC(=O)N2CC(CC(=O)OC)C2)CCC1 CCCCC(F)C(=O)N1CCCC(C(C)(C)C(=O)NCCOCC2CCCC2)C1 C1(NC(C2N(CC)CC2)=O)CC2CN(C(C3CCCN3C)=O)CC12 c1(CC)ccc(Br)c(NC(=O)CN2CCN(Cc3ccc(Cl)cc3C)CC2)c1 N1(C(C(F)=CC)=O)CCN(C2CCCN(C(c3nncs3)=O)C2)C(=O)C1 C12(C(=O)OCC(=O)Cc3ccc(O)cc3)CCC(CC1)OC2 C1(C(=O)OC)CC(O)CN1Cc1ccnc(-c2ccccn2)c1 c1(C(=O)OCC)cn(C2CN(C(C3(C)CC3C)=O)C2)nn1 C1(NC(Cc2c(C)ocn2)=O)CCC(CNC(c2cnc(O)s2)=O)CC1 C1(NC(c2cnn(CC)c2Br)=O)CCCC12CCN(C(=O)CNC=O)CC2 c1(C(N2CCCCC(NC(C3CC(=O)N(O)C3)=O)C2)=O)cc2cnccc2[nH]1 c1(OC)cc(F)ccc1CC(N1CC(O)CC1C(=O)Nc1cccc(CO)n1)=O c1(SC)cc(C(N2CCCC2CN(C)C(C2CCO2)=O)=O)c(Cl)cc1Cl CC(CNC(=O)C(C1CCC1)NC(c1ccns1)=O)CCCO Cn1c(CCC(=O)NC2CC(Nc3ncccn3)C2)nnc1S c1(OC)ccc(F)c(CC(=O)NC2CC3CC2CN3C(=O)C2=CCOCC2)c1 N1(C(C2C(OCC)C2)=O)CCN(C2CN(C(=O)C(C)Cc3c(C)noc3C)C2)CC1 C1(C)(C(=O)NCc2c(COC)cccc2)CC2CCC1CC2=O c1(OCOC)ccc(-c2ccc(NS(=O)(=O)CC#N)s2)cc1F N1(C(C(=Cc2cccs2)C)=O)CCC(C)C(NC(c2cn(C(C)C)cn2)=O)C1 C1(C(=O)NC2(CCCC)CC2)C(C)CCN1C(c1cccc(C)n1)=O C12(C(=O)NCC3(C)CCCN(C(C=CC)=O)C3)C3C4C1C1C2C3C41C(N)=O C1(NC(CN(C(C)C)C)=O)CCN(C(=O)C(C)(C)C(F)(F)F)CC12CCC2 Cc1cc2ncc(-c3nnc(N4CC(C)(C)CCC4(C)C)n3C(C)C)c(C)n2n1 C1(O)(CNC(c2ccn(C3CC3(F)F)n2)=O)CN(C(c2cn(CCF)nn2)=O)C1 Cc1c(F)ccc(Br)c1C(=O)NC(C)C(C)NC(=O)C=Cc1cnc[nH]1 C1(CC(=O)NC2CCCCC2NC(c2cc(C3CC3)cs2)=O)C=CS(=O)(=O)C1 C1(C(=O)NC(C)CCNC(c2csc(=N)[nH]2)=O)NC(=O)OC1C N1(C(c2cccc(CC=C)c2)=O)CCCCC(N(C(=O)C(CCC)OC)C)C1 n1(CC)ccc(C(=O)NCC2CN(C(=O)CSCC(=O)OC)CC2OC)cc1=O C1(C(N(C2(CO)CC2)C)=O)CC2(CC(NC(=O)CN3CC4CC4C3)C2)C1 N1(CCNS(C)(=O)=O)CCC(C#N)(C2(C#C)CC2)CC1 Cn1ncc2c1CN(C(c1cc3c(s1)CCC(C(C)(C)C)C3)=O)C2C(=O)O c1(C(=O)NC(C2N(C(C(CCC)C#N)=O)CCC2)C)c(Cl)sc2nnsc12 N1(C(C(=O)NCCOCC)CC2C3CC=CCC23)CCP(C)(=O)CC1 C(=O)(C1CCc2cc(OC)ccc21)NCC1N(C(c2n(C=C)ncc2)=O)CCC1 C(c1cc(C)cc(C)c1)=CC(=O)NC(C1(O)CN(C(COCCC#C)=O)C1)C C1(CNCc2c(C3CC3)cc(F)cc2Cl)COCC2(CCNC2)O1 C(=O)(C1=C(C#N)CCC1)NC1C(CC(=O)NC(C)CCN(C)C)CCCC1 c1(OC)c(C(=O)NCC2CCCN2C(c2nnc(C)s2)=O)oc2ccccc12 N1(C(C(=O)NCC)=O)CCN(C(C)C(N2CCCCC2)=O)CC1 c1(C(=O)NC2C(NC(CCC)=O)CCC2)cc(NC(=O)C#CC2CCC2)ccc1Cl c1(N2CCC(N(C(=O)CCCCCF)CCC)C2)ncn(C)c(=O)c1Br c1(C(=O)NC2CCC3(C(NC(=O)C=C4CCC4)C3)CC2)coc2c1C(=O)NCC2 c1(C(N2C(CN(C(=O)CNC(=O)C(C)(C)C)C)CCC2)=O)ccc(N)cc1F C1(C(=O)NCC2CC3CN(C(c4ncncc4Cl)=O)CC23)CCc2nc[nH]c2C1 N1(C(C(CC#C)O)=O)CCC(C(=O)N(CCCN(C)C)C)C1(C)C C1(NC(CC2(C)CCN2C(=O)Cn2cccc2)=O)CCCC(O)C1O C12(NC(=O)COCC3CCCC3)CCC(C1)N(C(c1c(N)cccc1F)=O)C2 Cc1ccn2c(CN(C3CCCC3)C(C)C(C3C(F)(F)C34CCC4)=O)cnc2c1 N1(C(C(C2CC2(C)CC)OCP(C)(C)=O)C(=O)NC)CC(CO)CC(C)(C)C1.CCO C#CC1(C(=O)NCCCCNC(C2CCNC2=O)=O)CCC1 CCCCC(O)CC(=O)NC1(CO)CN(C(c2ncc(C(=O)OC)cc2Cl)=O)C1 N1(C(c2c(C)nc(=N)[nH]c2)=O)CC(CO)C2(CCN(C(=O)C(F)C(C)C)CC2)C1 N(C(=NCC(C(F)(F)F)N1CCCC1)NC1CC(OC)C1(C)C)C1CCOC1 c1(C(=O)NCC(C(C)(C)C)NC(C=CC=CC)=O)cccc2c1OCCC2 C1(NC(C2(C)CCSCC2)=O)CS(=O)(=O)CC1NC(c1ncc(F)cc1N)=O C1(C(=O)C2CC2)CC=CCN1C(=O)Cn1cc(CCC2CCCO2)nn1 Cc1nc(=N)[nH]c(C)c1C(N1CCCCC1c1ocnc1C(=O)O)=O C1(NC(CCCCCCC)=O)COC2(CCN(C(=O)CC3CCOC3=O)CC2)C1 c1(OC)cc(C)sc1C(=O)NCC1CCCC1NC(=O)C=CSC Cc1ccc2cc(C(=O)NCC(C)NC(c3cc4ccsc4[nH]3)=O)ccc2c1 N1(C(CCn2ncc(C)c2)=O)CCC2(CCC(NC(=O)C(C)S(N)(=O)=O)C2)CC1 c1(C(=O)NCC2CC(NC(=O)C=C(Cl)Cl)C2)cncc(OC(F)(F)F)c1 N1(C(c2c(C)noc2)=O)CC2CCC1C1CN(C(=O)CSCC(N)=O)CC21 C(=O)(C1=C(Cl)CCCC1)NC1C(CNC(COc2ccc(OCC)cc2)=O)C1 N1(C(C2(C)CC2)=O)CCc2cccc(C(=O)NCc3ccc(F)nc3)c2C1 c1(C(N(CCN(C(c2c(CCC)nns2)=O)C)C)=O)cccn2cc(C)nc12 c1(CC(=O)NCC(c2cccc(Cl)c2)OC)cn(C)nc1I c1(NC(C2C(CNC(C=C(C)C(F)F)=O)CC2)=O)ccc(OCF)cc1 C1(C(=O)NC2(C(=O)N(c3cn(C)nc3O)CC)CC(OC)C2)CCCC12CCC2 n1(CCC(=O)NCC2CC2CNC(C2CCC(F)CC2)=O)ccc(O)nc1=O C=CC1(C(=O)NCC2CN(C(c3ccc(CC)o3)=O)CC2C)CCCC1 N1(C(C=C(C)C2CC2)=O)CCC(C(=O)NC(C)CC(F)(F)F)CC1(C)C Cc1cc(C(=O)N(C)CCNC(=O)CSc2nncn2C)nc(C(F)(F)F)n1 c1(CNC(Cc2nc(C)oc2)=O)nn(C)c2c1CN(C(c1cn(C)cn1)=O)CC2 CCC(C)C(C(=O)Nc1nocc1C(C)C)N(C1CC2(CC(OC)C2)C1)C c1(NC(CC(CC(C)C)O)=O)nc(Cl)nc2cc(Br)cnc12 C1(CNC(c2ccn(C)c2)=O)CCCCN(C(=O)Cc2cccnc2N)C1 CC1CN(C(c2cc(C(F)F)nn2C)=O)CC(C)C1NC(=O)Cc1csc(=N)[nH]1 C(=O)(C(C(C)C)N1CCCC1)NCC1(OCC)CN(C(=O)C(F)OC(F)(F)F)C1 CCCCCCCCC(=O)NCC1(C)CCCN(C(c2cnccc2CC)=O)C1 Cc1ncnc(C(=O)NCC2CCC2NC(=O)CCSc2ccccn2)c1C CC(C)C(C)C(=O)NC1CN(C(c2csc(C(F)F)n2)=O)CC1C N1(C(CCCCC#C)=O)CCC2CCN(C(c3cc(Br)ccc3C)=O)CC12 Cc1c(C(N2CC(CO)(NC(C3CC4(CC4)CO3)=O)C2)=O)nn(C)c1N Cc1cc(O)ncc1C(N1CCCC(N(C(=O)COc2ccon2)CCO)C1)=O C1(CNC(c2c(OCC)nc(C)cc2)=O)C2CCC1CN(C(=O)C(CC)CC)C2 CC1CC(NC(=O)CC2CCCCC2)CN(C(c2ccnc(C(F)(F)F)c2)=O)C1 N1(c2nnc(COCC)n2CC(c2ccccc2Cl)O)CCn2nccc2C1 C1(C(=O)NCCOC(C)=O)(NC(CCC)=O)CC1(C)C C(C)(CCCC(=O)NC1CN(C(c2ccc(O)cc2)=O)C1)c1ccc(OC)cc1 Cc1nn(C)c(=O)c(-c2nc(CCc3ccccc3)nn2CC2CC2)c1C c1(CC)cncc(CNC(=O)CNC(=O)CNC(C2CC23CC3(F)F)=O)c1 c1(C(N(C2CCN(c3snc(CC)n3)C2)C)=O)cnn2c1CCC2 C(C(C)(C(=O)NCc1cccc(O)c1)NC(=O)C(C)C)SC CN1CCC(C(=O)NC2CC(N(C(=O)C=Cc3cscn3)C)C2)C1 C#CCC(CC(F)F)C(=O)NCC1C2CN(C(c3nccn3C)=O)CC12 c1(C(N2CC(NC(c3ccc(O)nn3)=O)C3C2C3)=O)cc2nccnc2cc1F c1(OCC(=O)NC(CCCNC(CC=C(C)C)=O)C)cccc([N+](=O)[O-])c1 c1(C(=O)NCCN(C)C(C2CC2c2cccs2)=O)cnc(N(C)C)s1 C12(NC(C(CNC(C(C=C)C)=O)N(C)C)=O)CCC(CC1)C2(C)C c1(CNC2CCC(NC(=O)CC3CCC(C(=O)O)CC3)C2)cc(F)c(F)cc1O C1(C#N)(C(=O)NC2C(NC(Cc3cn(C)nc3)=O)C2)CCS(=O)(=O)CC1 C(=O)(CCCN(C)N=O)NCCCC1CCN(C(C2CC(C#C)(O)C2)=O)CC1 c1(NCCNC(C2CCCCCC2)CC)ccnc(C)n1 C1(OCCn2cc(CNC(C3N(C(C)=O)CCC3)=O)nn2)CCCN(C(N)=O)C1 c1(C(C)C)ccc(S(=O)(=O)N(C2CCN(S(=O)(=O)c3cnn(C)c3)CC2)C)cc1 C12(CNC(=O)C=Cc3ccco3)CCCCC1CN(C(c1cnsn1)=O)C2 n1(CC(=O)OC)ccc2c(NC(C3CC(F)(F)CC3N)=O)ncnc12 C(=O)(C(CO)NC(=O)C(c1cccnc1)N)OC c1(NC(c2ccc(C(C)CC)cc2)c2n(CCCC)nnn2)cccc(C#N)c1 c1(C(=O)NCC(CO)NC(CCCOC)=O)cnc(C2CCC2)nc1O N(C1CCCn2ccnc21)C(CC(CNC(C1(C)CC(F)(F)C1)=O)OC)=O C1(NC(Cc2[nH]c(=N)sc2)=O)C2CC(O)C1N(C(=O)Cn1nc(Cl)ccc1=O)C2 C12(CNC(C3(CC)CC3)=O)CC(CO1)N(C(=O)Cc1ccccc1CO)C2 C1(CC)C(=O)NC(C2CC2)C(=O)N1.C(C)(C(=O)OCC)SCCCC C(=O)(CCN(OC)C(=O)C1(C)CCCN(C)C1)NCC#CC CC(C)CS(=O)(=O)CC(=O)NCCN(CC(C)O)C(c1ccc(=O)n(CCF)n1)=O C(=O)(C(CN(C)C)C(C)C)NC(c1nc[nH]n1)CC.C123CCC(CC1)(C2)NC3=O C1(C(N2CCC(O)(C(C)NC(C3CC(F)C3)=O)C2)=O)CCc2ccnn2C1 C1(C(=O)OC)CCC(C)N(C(c2nnc(NC(c3nc(Cl)ccc3Br)=O)s2)=O)C1 C1(NC(C(CCNC(C23OCCC(C)(C2)C3)=O)O)=O)CCCCC12CCC2 c1(C(C(=O)NCCN(C(=O)C=Cc2ncc[nH]2)CC2CC2)O)ccccc1Br C(C(C(=O)N1CC(Oc2ccccc2)C1)NC(N)=O)N(C)C1CC1.C1(O)CC1 c1(CNCC(CC(C)C)(C)C)nc(Br)n2c1COCC2 N1(C(CCN(c2ccccc2)C)=O)CC2CC1C2NC(c1c[nH]c(C(N)=O)c1)=O C(=O)(C(CC(C)C)c1ccc(Cl)cc1)NC1C(NC(c2c(OC)cncc2)=O)C1 C=C1CON(C(=O)CC2CCCN(C(c3c[nH]c4ccccc34)=O)C2)C1 CN(C)NC(=O)CCC(=O)N1CCCC1C(C)(C)C(=O)NC1CC(O)C(O)C1 C1(NC(CC2CCN(C(c3cncc(CC)c3)=O)C2)=O)CC2CCC(C1)N2CC C(=O)(CC(CC)C(C)(C)C)N1CCC(OCC2CCN(C(CCSC)=O)CC2)C1 C(CC(C)(C)C)(C(=O)NCc1ccc(F)cc1)NC(CCCOC(C)=O)=O Cc1nnc(CCC(=O)NC(CO)C(C)NC(=O)CC2CC2(C)C)n1C C1(CNC(C2N(C)C(=O)NC2)=O)CC2COCC2N1C(c1csc(Cl)c1)=O CCCCCC(O)CC(=O)N1CCC(CNC(c2ccc(Cl)cn2)=O)C12CC2 c1(CNC(C)Cc2ccccc2Cl)ccc2nc[nH]c2c1 Cc1cnc2n1CC(C(=O)NCC1CCC(CNC(=O)C(C)CO)CC1)CC2 Cc1cc(C(=O)NCCC(C)NC(=O)CCCN(C)C(=O)OC(C)(C)C)sc1Cl Cc1cccc(C(=O)NC(CNC(C2CC3CCC2O3)=O)CC(C)C)c1 c1(C(N2C(CNC(C=CS(C)=O)=O)CC(O)C2)=O)cccc(Br)c1F Cc1ccc(F)c(S(=O)(=O)NCCC(=O)NC2CC2CNC(=O)CN(C)C)c1 S(=O)(=O)(CCC(=O)NC1(C)CC(NC(=O)CC2CC3CC3C2)C1)NC C1(C#N)(OC)CC(C(=O)NCC(C2CC2)NC(c2cc(C)oc2C)=O)C1 S(=O)(=O)(c1ccc(NCC2CCCSC2)cc1Br)N(CCC#N)CC1CCCO1 c1(CC)ncc2c(n1)CCN(c1cc(N3CCN(c4cccs4)CC3)ncn1)C2 C1(C)(C(=O)NCC2(CC(=O)NC3(C(COC)O)CC3)CC2)CC=CCC1 C(CC(C(=O)NCCCC1(O)CC1)NC(c1cnc(S)nc1)=O)N(C)C N1(C(c2ccc(C=C)cc2)=O)CCN(N(C(C)(C)C)C(C)C)CC(C)C1 c1(C(N2CC(CNC(c3c(CC)nns3)=O)C(C)C2)=O)c([N+](=O)[O-])c(C)nn1C c1(C(=O)NC(CC)(C)CCC(=O)O)nc2ccccc2n1C1CCN(C)CC1 N1(C(C(C)(C)CF)=O)CCC=C(C(=O)NCC2CCOC2C(=O)O)C1 C(=O)(C(CNC(=O)C(CN(C)C)N(C)C)CC1CC1)NCCNC(C(C)C)=O C(=O)(CC(C)CC(F)(F)F)NC1C2(CN(C(c3c(C)cccc3F)=O)C2)CCC1 C#Cc1cccc(C(=O)NC2CC(C)(NC(c3cc(C)nc(C)c3)=O)C2)c1C N1(CC)CC(C(=O)NCC2CCC(F)(CNC(=O)C(C)(C)CO)CC2)CCC1=O c1(OC)ccccc1CC(C)CC(=O)NCC1(NC(=O)CCN(C)CCO)CC1 c1(C(N2CC(C(=O)Nc3cn(CC)nc3)C(C)C2)=O)c(F)ccc(OCC)c1N c1(C(c2n(CCSC)nnn2)NCC(C)(CC)C(C)O)ccc2occ(C)c2c1 C(=O)(C(CC(N)=O)NC(=O)CC1(C)CC1)NC1CCC(C(=O)OC)C1 N1(C(CC(CC)C)=O)CCCC2(C1)CN(C(=O)C(C1CCC1)OC)C2 C(=O)(CCC(C)(C)[N+](=O)[O-])N(CCCCCCNC(=O)CCCCC1CC1)C S(=O)(=O)(c1cccc2c(Cl)nccc12)N1C2CCN(C(CC)=O)CC2CC1 C1(NC(c2cc(CNC(c3ncccc3Cl)=O)no2)=O)CC2CCC1O2 c1(C(=O)NC2(C(N(C)Cc3nc(C)on3)=O)CC2(C)C)cccnc1S c1(OC)ccc(C(=O)NC2CN(C(c3cnn[nH]3)=O)CC2O)nn1 c1(C(=O)NCC(C2CCCC2)NC(CC2(C)CC2(Cl)Cl)=O)cccc(C2CC2)c1 C(CCNC(C1CCCCC1n1ccnc1)=O)(C(C)C)NC(c1cc(C)[nH]n1)=O N1(C(C(COC)(F)F)=O)CCC(C)(C)C(CNC(C2(SC)CC2)=O)C1 c1(NC(c2scc(-c3cc(OC)c4c(c3)OCO4)n2)=O)nc(Cl)ccc1[N+](=O)[O-] C(=O)(C(F)C(F)(F)F)NC(c1nc(C(F)(F)F)cs1)C(=O)OC N1(C(C2(CC=C)CCC2)=O)CCCC(NC(=O)CC(CC)C2CC2)C1 c1(CC)ncc(Cl)c(C(=O)NCC2(F)CN(C(=O)CN3CC(C)(C)C3)C2)n1 Cc1ccc(C(=O)NC2CC(NC(=O)CSc3ccccn3)C2)c(Cl)c1C C1(C)(NC(C(C=C)O)=O)CCN(C(c2cc(C(C)C)nn2-c2ccccc2)=O)C1 c1(C(=O)NC2C(OC)CN(C(=O)C(c3cnn(C)c3)O)C2)cc2c([nH]1)CCOC2 CN=c1nc(N2CCC(C)(N(C)C)C2)[nH]c(=NCC2(F)CCOCC2)[nH]1 N1(C(=O)OC(C)(C)C)CC2CCCC2(c2nc(NC(=O)COCC3CC3)no2)C1 c1(C(=O)NC2(C)CC(NC(C(C)O)=O)C2)ccc(=N)[nH]c1 CCCCC(CNC(=O)CN(C(=O)C(c1cccn1C)=O)CC)CCC C(=O)(CC1OC(=O)c2ccccc21)N(C)CCN(C)C(C1Cc2cscc2C1)=O C(=O)(C1=CCS(=O)(=O)C1)N1CCN(C(C2CC3C(C2)C3(F)F)=O)CC1CCO N1(C(c2c(C)c(Br)cnc2)=O)CCN(C(=O)C(C)(C)F)CC2(CC2)C1 N1(C(=O)NC2C(C)COC2)CCc2nc(O)ccc2C1 C(=O)(C1=CC2(CCN(C(=O)C(C)n3ccnn3)C2)C1)N(c1ccc(CC)nc1)C C1C(C)(C)C(=O)N1.C=CC(O)C(=O)NC(CC1CC1)C(=O)OC C(=O)(C(O)C(C)(C)C)N1C(CNC(c2nc(OC)oc2)=O)C=CC1 O=S(=O)(NCC(O)COc1ccc(Br)cc1)N1CCc2ccccc2C1 N1(C(c2cnc(C(C)OC)s2)=O)CCN(C(C23CC(F)(C2)C3)=O)C(CO)C1 N1(C(CCC=C)=O)CC2(COC(CNC(=O)Cc3nocc3C(C)C)C2)C1 C(C(C)C(C)(C)C)N(C(c1snc(OC)n1)c1ccccc1)C c1(C(N2CC(NC(c3cc(O)cc(F)c3)=O)C(F)CC2)=O)ccc2nc[nH]c2c1 C1(C(=O)NC(CC)(C)CO)C=CCN(C(=O)C(=C2CCCCC2)F)C1 C(C(=O)N1CCN(C(C)CNC(=O)C=Cc2cocn2)CC1)(C(C)C)SC Cc1cn2c(CC(N3CCN(C(=O)C4=CCCCO4)C(C)C3C)=O)csc2n1 c1(C(=O)NCC2(C)CCN(C(=O)Nc3cc(F)ccc3F)C2)ccc(O)cc1Cl C(=O)(CCCCN(C)C(C)=O)N(CCNC(c1cnc(CC)s1)=O)C c1(C(N(C2CCN(C(c3cc(Cl)c(Br)c(Cl)c3)=O)C2)C)=O)ccc2c(c1)OCO2 N1(C(C(C)=C(CC)C)=O)CCCOC(CNC(=O)CC2CCN(CCF)CC2)C1 C1(=O)CCCCN1.c1(CONC(CC2N(CC)CCC2)=O)ccccc1F c1(C(N(CC(O)CNC(c2ccoc2Cl)=O)C)=O)cc2ccc(F)cc2nc1O NC1CN(C(c2cc(Cl)ncc2F)=O)C2(CCCCCC2)C1 Cc1ccc(NC(C2CCCCC2OCc2ccccc2)=O)cc1-c1nn[nH]n1 N1(C(C(CC=C)C(C)C)=O)CC2(C1)CN(C(=O)COCc1ccccc1)CCO2 N1(CC)CCCC1C(=O)N(C)CC1(NC(=O)CC2CCCO2)CC1 C(=O)(CCC(C)(C)C#N)NC(CN(C(C1CC1c1ccncc1)=O)CC)C C(C(=O)NCc1cc(Cl)ccn1)(C(C)O)NC(C=CCCC)=O C1(NC(CC=C=C)=O)(CNC(=O)C(C)(C)CN2CCN(C)CC2)CCCCC1C N1(C(c2c(C)con2)=O)CC2CN(C(c3cc(Br)ccc3N)=O)CC2C1 C(CC(O)CN(C)C(c1ccc(CN(C)C(=O)OC(C)(C)C)o1)=O)OC Cn1c(C(N2CC3CC2CN3Cc2c(Cl)cncc2Cl)=O)cccc1=O Cc1c(C(N2CCCC2CN(C(=O)C#CC(C)(C)C)C2CC2)=O)cncc1Cl N1(C(C2C(COC)CC2)=O)CCC2(CCCN(C(=O)CSc3cccnc3)C2)C1 C#CC1CN(C(c2cn3ccnc3cn2)=O)CCN1C(C1CC1C(C)(F)F)=O CC1(CC(=O)NC2(CCO)CN(C(C3(C(N)=O)CCC3)=O)C2)OCCO1 Cc1cc(C(=O)NC2COCCC2NC(C2CC23CC(F)(F)C3)=O)c(Cl)cc1N c1(N2CCC(NCCC(N3C4CCCC3CC4)=O)CC2)cccc2c1OCCO2 CCC(C)CCCC(=O)NCC(C)(C)NC(c1cn(CCOC)nc1C)=O c1(C(=O)NC2CCN(C(CCC=C)=O)C(C)C2)ccc2c(c1)C(=O)CCC2(C)C C12(CNC(COCC(=O)OC)=O)CCCC1CN(C(C1(C)COCCO1)=O)C2 N1(C(C2C(CC)CCC2)=O)CC(F)(F)CC1(C)CNC(c1snnc1C1CC1)=O C(=O)(C(=O)N1CCC(O)CO1)NC(COC(C)C)C c1(C(N2C(CNC(C(C)NS(C)(=O)=O)=O)CC2)=O)cc2sccc2cn1 C1(N(C(c2nnc(CC)s2)=O)C)CC2CCC(C1)N2C(C1(OC)CS(=O)(=O)C1)=O c1(OC)cc(C(N2CC(=C(F)CNC(=O)C(c3ccccn3)C)C2)=O)nn1C n1(CC)ncc(Cl)c1C(N1CCC(C(C)NC(C2(C#N)CC2(C)C)=O)CC1)=O c1(C(=O)NC23CCN(C(CS(CCC)(=O)=O)=O)CC2C3)nc2nccc(C)n2n1 C1(CC)C(NC(=O)CN(C)S(N)(=O)=O)CCN1C(c1cn(C2COC2)nn1)=O C1(C(=O)NCC(C)(O)C2(C)CC2)(SC)CN(C(=O)C(F)OC(F)(F)F)C1 c1(C(=O)NC2CN(Cc3ccc(OC)s3)CC2O)cnc2ccccn12 c1(OC)ccc(C2CC2CC(=O)NC2CCCC2Oc2ccc(Cl)cc2)cc1 N1(C(C2(CNC(CC3CC(=C)C3)=O)CCCCC2)=O)CC2CN(C)CC2(C)C1 N1(c2nc(NCC(=C)Br)c3c(n2)scc3)CCc2c(Cl)cc(F)cc2C1 Cc1coc(C(=O)NCC(C)CNC(c2cc(-c3cnn(C)c3C)no2)=O)c1C C1(CC(=O)N(CC#C)CC2CC2)CC(NC(c2cc(O)nn2C)=O)C1(C)C C(=O)(C1=NOC(C)(C)C1)NC(CN(C(c1scnc1Br)=O)CC)C C12(NC(Cc3cccc(C)c3)=O)CCCC1N(C(c1ccc(F)cc1Cl)=O)CC2 c1(CC(C)C)ccc(C(=O)N(c2ccc(N(C)C)nc2)C(C2C=CC(N)C2)=O)cc1 c1(C(=O)NCC2CCN(C(C(C)N(C)C)=O)C2)c[nH]c(=NCC(F)(F)F)cn1 c1(C(=O)NCC(CO)NC(C=CSC)=O)cnn(C)c1C(F)(F)F C1(NC(CONC(CNC(=O)OCC)=O)=O)CN(C)CC1(F)F C1(CC(=O)NCCCC(O)CO)CC2(C1)CN(C(C1(F)CCOC1)=O)C2 c1(C(=O)NC2C(NC(c3nc(C(=O)OC)oc3)=O)CCCC2)c(C)[nH]c(C)c1C c1(C(=O)NC2CCN(C(C(CC)CCOC)=O)C2(C)C)cn2c(C)cccc2n1 Cc1nc(NCC23CC(CN2C(C2CCCCN2C)=O)C3)cc(O)n1 c1(C(N2CCC(NC(=O)CCC3OCCO3)(CO)C2)=O)ccn2c(O)nnc2c1 c1(C2C(C(=O)OC(C)(C)C)C2)ccc(NC2CCCC2O)cc1 Cc1cccc2oc(C(=O)NC(C)CC3CCN(C(=O)C(C)N(C)C)CC3)cc12 C1(C(=O)NC(CCNC(C(C=C)OC)=O)(C)C)CCOC1C=C C1(C(=O)NCc2scc(C(=O)NCC3(C)CC3C(F)(F)F)c2)OCCC1(C)C CC(c1ccc(C(F)(F)F)cc1)=CC(N1CCC(NC(=O)CC(C)(C)SC)C1)=O c1(NC)nc(NCC(=O)NC(c2cc(F)cc(Cl)c2)C2CC2)c2ncsc2n1 c1(CCC(=O)NC(CNC(C2(CCOC)CCCC2)=O)C)ncc(F)cn1 c1(CN(C(=O)CCOC(CN2CCCC2)=O)CC)cccc(NC(C)=O)c1 C1(C(=O)NC2CC(N(C(C(C)Cc3cnco3)=O)C)C2)CC12CCCCC2 N1(C(c2ccc(C)c(OC)c2)C(=O)NCCC2(C)CC2)CC2CCN(C)CC2C1 N1(C(c2cnn(C(C)C)c2F)=O)CCCC12CCN(C(=O)C=CCO)C2 c12nc(cs1)C(=O)NCCN2C.CC(C)C(=O)NCC=CCNC(c1nc[nH]n1)=O c1(C(=O)NC2C(NC(C3N(CC)CCOC3)=O)CCC2)n[nH]c2ccc(Cl)cc12 NC1CS(=O)(=O)CC1NC(c1c(Cl)cncc1Cl)=O C#CC1(NC(=O)C(C)C(C)NC(c2cc(C)nc(C)n2)=O)CCCCCC1 C1(NC(CC2N(C(c3nc(C)sc3)=O)CC2)=O)CCCC2(CC1)CC2 c1(SC)ccnc(N2CCC(NC(c3ccnc(O)c3)=O)C2)n1 C(=O)(C(O)C(C(C)C)OC)NC1CCN(C(c2ccc(C#C)cc2)=O)C1C(C)C N1(C(CNC(=O)Nc2c(C)cccc2)=O)CCN(C(=O)C(C)N(C)C)CC(O)C1 c1(C(=O)NCC(CC)NC(=O)CSc2cccc[n+]2[O-])cn2nc(C)sc2n1 CP(C)(=O)c1ccc(C(=O)NC2CC(CNC(C3CC4COCC4C3)=O)C2)o1 N1(C(C=CC2(C)COC2)=O)CCC2CN(C(=O)CCC3CCCO3)CC12 CCC(N=c1[nH]c2c(c(=NCCCC#N)[nH]1)SCC2)c1ncc[nH]1 C1(CC(=O)OCC(=O)N(CC=C)C)CCC(=O)N1 C1(CNC(c2c(C)n(C3CC3)nc2)=O)CCN(C(=O)Cc2cn[nH]c2)C12CCC2 c1(OC)ccc(O)cc1-c1csc(C(=O)N(CC#N)Cc2ccccc2)n1 CC1(C)CC(C(=O)NCc2csc(CNC(c3cc(C4CC4)no3)=O)n2)CO1 N1(C(C2C(OC)CCCC2)=O)CC2(C1)CN(C(c1coc(C)c1)=O)CCO2 C1(C(=O)NCC2(C(C)NC(c3c(C)csc3)=O)CC2)CCC(C(F)F)CC1 C1(NC(c2ccc(C3CC3)o2)=O)CCCCCC1NC(C1CSCCS1)=O C1(NC(CCS(=O)(=O)NC)=O)CCC2(CCCN(C(c3cc(OC)cs3)=O)C2)C1 c1(CNC2C(C(N3CCN(C)CC3)=O)CCC2)cccc(F)c1Cl C(c1ccccc1)=CC(N1CC=CC(NC(C2(CF)CC(F)(F)C2)=O)C1)=O c1(OCC(N2CCN(C(C3C(C4CC4)C3(F)F)=O)CC2)=O)cccc2nsnc12 N(C(=NCCCC(C)(C)C)N1CCC2CCCCC2C1)CC(C)C c1(C(N2CC(O)CC(NC(C3(N=[N+]=[N-])CC3)=O)C2)=O)ccc2c(c1)CCOC2 c1(C(=O)NC2CC(O)(CNC(c3c(C)n(C)cn3)=O)C2)ccc(O)nc1Cl c1(C(N2CC(F)CC(C(=O)NC(C#C)C)C2)=O)cc(O)cc([N+](=O)[O-])c1 c1(C(=O)NC2C(CNC(c3ccnnc3)=O)CC2)nc2ccc(Br)cn2n1 C1(C(N2C(Cn3cc(-c4ccc(C)cn4)nn3)CCC2)=O)CC12CCCCCC2 C(C(C(F)(F)F)N1CCN(C(C2CCCCS2)=O)CC1)NC(COC)=O c1(CC(=O)NCCNC(c2ccc(C#C)cn2)=O)cccc2c1CCC2 C1(CNC(C2C(=C)C2)=O)CCC2(CCN(C(c3cnc4n3CCS4)=O)CC2)CO1 N1(C(C=C(C)Cl)=O)CCCN(C(=O)CCc2ccnc(Cl)c2)C(C)C1 C1(C)(NC(c2c(CNC(Cc3cc(CC)no3)=O)noc2)=O)CCCC1O N1(C(c2c(C)cns2)=O)CCC(C)(CNC(c2ccc(O)c(N)c2)=O)CC1 c1(C(=O)NCCC(CNC(C2(CCC)CC2)=O)O)[nH]cnc1C#N N1(S(=O)(=O)c2cccc(Cl)n2)CCc2cc(-c3ccc4nonc4c3)cnc2C1 c1(C(N2C(CNC(C3C(C)=C3)=O)CC3(CC3)C2)=O)cnn2c1NCC(C)C2 C1(CNC(c2ncnc(OC)c2F)=O)(CO)CC12CCN(C(=O)C=C(C)C)CC2 N1(C(C2(OC)CCC2)=O)CCCCC(C2CN(C(C34CC3CCC4(F)F)=O)C2)C1 CCCS(=O)(=O)C(C)C(=O)N1CC(NC(c2cccc3[nH]ncc23)=O)CCC1C CC(C)(C)C1=NOC(C(=O)NCCCNC(=O)CCCN2CCCC2)C1 C1(C(=O)NC2(C)CCOC2=O)(CC)CCN(C(C2CN(C)CCO2)=O)CC1 CCC(COC)C(=O)N1CC(CCNC(C2(O)CCC2)=O)(OC)C1 c1(C(N2CC(C)C(NC(C3CCC(=O)N3)=O)CC2)=O)cccc(N=[N+]=[N-])c1 CCCCC(C(=O)NCc1csc(CNC(=O)COC(C)C)n1)ON=C(C)C CC1CCC(F)(C(N2CCN(C(c3sccc3F)=O)C(CC3CC3)C2)=O)CC1 C#CCC(C)(CNC(=O)NC1(Cc2ccccc2)CCOC1)CO N1(Cc2nnn(C)n2)CCCCC1CNC(=O)CC(=O)Nc1cccs1 c1(C(=O)NC(CN(C(=O)C(O)Cc2cn(C)cn2)CC)C)ccn(C)c1 c1(C(N2CC3CN(C(=O)C(Cl)(Cl)Cl)C3C2)=O)cc(I)c(F)cc1F N1(C(C(N=S(C)(C)=O)=O)=O)CCC(C2CC2NC(c2sccc2Cl)=O)CC1 C1(NC(=O)Cc2ccco2)CCCN(C(=O)CCc2cccc(F)c2)CC1 c1(C(N2C(C)CC2C(N2CC(F)(F)C2C2CC2)=O)=O)cn2ccccc2n1 C1(NC(c2ccoc2C(F)(F)F)=O)CN(C(C2CC2CF)=O)CC12CCC2 c1(N2CC(CCCCNCc3ccc(N(C)C)cn3)C2)nc2cccc(F)c2o1 c1(C(=O)NCCCC(=C)C)ccc(C)c2c(C#N)c[nH]c12 N#Cc1ccc(Br)cc1CN1CC(C(=O)Nc2ccc(F)c(I)c2)C1 c1(C(=O)NCc2cccc(CNC(CC)=O)c2)cnc2nc(C)ccc2c1O c1(CC(=O)NC2CC(F)(CNC(CC(C)C)=O)C2)cnn2ccccc12 c1(-n2cc(C3(F)CN(C(CCOCCC)=O)C3)nn2)cc(Cl)c(Cl)cc1Cl Cc1cncc(CC(=O)NC(C)CCNC(c2onc(C)c2C)=O)c1 C=C1CCN(C(C2(C)CN(C(c3scc(C)c3Cl)=O)C2)=O)CC1 C(=O)(C1=NN(CC)C(=O)CC1)N(CC(CC)NC(c1ccn(C)c1)=O)C C1(CNC(c2ccc(C)o2)=O)CCC(C)(C)CN1C(=O)CCCCc1cnc[nH]1 CC1OC2(C(=O)NCC3(c4ccc(C(=O)O)cc4)CC3)CCC1C2 C1(C)(COC)C=CCN1C(=O)CC(CC1CC1)NC(c1nnn(C)c1C)=O C1(NC(c2nnn(CC)c2C)=O)(CNC(=O)C(F)=C2CCC2)CCCCC1C CCC(CCC(=O)NCCCC1(O)CC1)NC(=O)CC(C)C1CC1 C1(CCC)CN(C(c2sc(OC)nc2Cl)=O)CCN1C(=O)CP(C)(C)=O CC1(C)CN(C(C2(O)COC2)=O)CC2(CN(C(=O)C(C3CC3)C3CC3)C2)O1 N1(C(C(C)NS(C)(=O)=O)=O)CC2CCCN(C(=O)CCC3CCCC3)C2C1 c1(CC)cncc(CO)c1.C12(C(=O)NC(=O)CSCCN)CCCC1C2 c1(OC)ncc(C(N2CCC(NC(c3cc(C)co3)=O)C23CC3)=O)nc1C C1(C(N2C(CNC(c3c(OC)ccc(C)n3)=O)CCC2)=O)CCn2ccnc2C1 c1(C(=O)OCC)ccc(Cl)cc1S(=O)(=O)Nc1nc2cccc(C)c2s1 c1(N2C3(CN(c4nc(SC)nc(C)c4Br)C3)CC2)ncc2cccc(Br)c2n1 C1(CC(=O)NC(CCNC(CCCC(C)C)=O)C)CCc2sccc2C1=O c1(C(=O)NC2CN(C(c3ccncc3)=O)CCC2CO)cc2c(=O)cc[nH]c2s1 c1(NC(C(C)=CC=C)=O)cnn(CCOC)c1C.N12CCCC1CC2=O C1(CNC(CC2N(C)CCOC2)=O)CCCCN(C(c2cn3c(n2)CCC3)=O)C1 c1(CN2CCCC(N)(CC)C2)nc2cccc(C)c2o1 C=CC(CC)CC(=O)N1CCC(OCC(N2CC(SC)C2)=O)C1 CCCC(C)(C)C(=O)N1CC2C(CN(C(=O)CCc3ccccc3OC)C)C2C1 c1(C(=O)NC2CN(C(=O)CN3CCNC3=O)C3CC23)ccc(CO)c(Cl)c1 CCC(C)CC(=O)C(=O)N1CCCC1C(C)(C)C(=O)Nc1cncnc1O CCCCN=C(NCc1ncnn1CC)NC1CC(C)CC(C)C1 c1(C(C(=O)NC)N(C(C)C(=O)OC)C2CC2)ccc2c(c1)OC(C)(C)O2 C1(C(=O)NC(CO)CCF)(NC(C(c2ccnn2C)C)=O)CCCCC1 C1(C(=O)NCC(C)NC(C(CCC)OCC)=O)CCCN2CCCCC12 CC1(C)C(NC(=O)C=Cc2cccc(F)c2)CCN1C(c1n[nH]c(=N)s1)=O CC(CNC(=O)Cc1ccc([N+](=O)[O-])cc1F)N=c1ccnc(CO)[nH]1 C=CCCCC(C(=O)N1CCC(N2CC=CC2)C1)NC(c1cccnc1S)=O CN1C2CCC1CC(C(=O)NC1CC(CNC(=O)CN3CC(=O)NC3=O)C1)C2 c1(C(CNC(NNC(=O)c2ccc(C)s2)=O)=O)ccc(S(N)(=O)=O)cc1 N1(C(CCCc2onc(C(C)C)n2)=O)CCCC(N(C)C(c2cnccn2)=O)C1 C(=O)(CCCCCCC(C)C)N1CCC(C)(Nc2ccnc(C(CC)C)n2)C1 C(=O)(C(C)(C)C(C)(C)C)NCCOCCNC(C(C1CC(F)(F)C1)OC)=O c1(-c2cn(CCCC(=O)N3CC(C(c4cccnc4O)=O)C3)nn2)ccc(O)nc1 c1(C(=O)NC2CC(C)(NC(CC3C(C)CCC3)=O)C2)cnc2n1CCCC2 c1(NC(C(c2ccc(C(C)=O)cc2)CC)=O)ccc(C)c(SC)c1 c1(OC)noc(C(N2CC(CNC(=O)Cc3n[nH]c(C)n3)C(C)C2)=O)c1Br c1(OCCC(=O)NC(CC)CNC(=O)CSCCC#N)cccc(C)c1 c1(Cc2cn(C)nc2)nc(=NC(=O)C2(C)CNC(=O)N2)s[nH]1 CC(C)CCC(=O)NC(C)(C)COCCCNC(c1cnn(C2CC2)c1Cl)=O n1(CCCC)ncc(C(=O)NC(CO)C(C)NC(C2(C)CCCOC2)=O)c1C c1(N(C)Cc2cccnc2)nc(N2CCC3(CC2)CC3)nc2c(F)cccc12 c1(C(N2CC(CNC(CCCC#C)=O)C(C)C2)=O)cc(C#N)ccc1C C12(CNC(C(c3ccccc3)SC)=O)CN(C(=O)CCC3CC3)CC1CCO2 C=C(C)CN=C(NCC1CCCN1CC)NCc1ncnn1Cc1ccccc1 C1(C(=O)Nc2ccc(OC)c(C)c2)CN(C(C2(CO)COC2)=O)CC1C1CC1 c1(C(N2C(CO)CCC23CCC3)=O)cccc2c1OCC2 C(=O)(CC1=CCCCC1)O.c1(N(C(C)C)C)nnc(C2CCS(=O)(=O)C2)n1CC1CC1 C12(CCC(=O)NCC(CN(C(=O)C=CCO)C)(C)C)CC3CC(CC(C3)C1)C2 c1(C(=O)NCC(C)CN(C)C(C23CC(F)(C2)C3)=O)cnc(C2CCOCC2)s1 N1(CC)CCC(c2nnnn2C2CC2)(NCCCNC2CCCC2)C(C)C1 c1(N(C2CCNC2)C(c2nccc(C)c2)=O)ncnc2cccnc12 C(=O)(CC(O)CNC(C12CC(CO)(C1)C2)=O)N(C(CC(=O)OC)C)C C(=O)(C#CC1CCOC1)NC1CC(C)(NC(=O)Cc2ccc(Cl)s2)C1 CC1CCC(NC(=O)C(=O)NC2CCC3(CCC3)CC2)c2ccccc21 C(C)(C(=O)NC(C)CN(C)C(C)C)(C1CN(C(CC2C(CC)C2)=O)C1)OC c1(C(=O)NC2CC3(CC(C(=O)NC(C(C)C)CO)C3)C2)cc2ccccc2n1C C(C(=O)NC1CC(NC(=O)Cc2cn(C)cn2)C1)(C(C)C)OCC Cc1ccc(=O)n(CC(N2CC(NC(=O)Cn3nnnc3C)C(C)C2)=O)n1 C1(NC(c2ccnn2C(F)F)=O)CCN(C(C2CCC=CCC2)=O)CC1 c1(OC)c(F)cc(CC(N2CC3C(C(=O)NC(C)C#N)C3C2)=O)cc1F C=C(C)CC(C(=O)N1CCC1C(N1CCCC(COCC)C1)=O)OC c1(OC)c(C(=O)NCC2CCN2C(=O)C(C(C)O)NC(C)=O)csc1C N1(C(c2ccc(SC)o2)=O)CCC(F)C(NC(c2cn(C(F)(F)CO)nn2)=O)C1 CC(C)CC(C)(O)C(=O)NC1CCN(C(c2c(O)cc(Br)cc2F)=O)C1 c1(C(=O)NCCC2N(C(C(CC)C(C)C)=O)CCC2)cc(C)nc2c1cnn2C c1(C(N2CCCC(NC(=O)CC3CCCCO3)CC2)=O)nc[nH]c2ncnc1-2 Cc1nc(C2CC2)oc1C(=O)NCCOCCN(C)C(C1C(C)C1C)=O C1(C(=O)NC2CCC(CNC(C(C=C=C)C)=O)C2)CC2(CCOCC2)C1 c1(C(=O)NCC#CCNC(C2CN(C)C(=O)C2)=O)ccnc2ccnn12 C1(O)(C(C(=O)N(CCCNC(=O)CC2CCOC2)CCC)F)CCCC1 c1(OCC(=O)NCCCC(CO)NC(=O)CC2CCCSC2)ccc(F)nc1 C1(CC(=O)N(CCCN(C(=O)C=C2CCC2)C)C)CC(=O)c2ccccc2C1 Cc1cc(O)cc(C)c1CC(=O)NC1CCC1NC(=O)C(C)C CCC(C)C(C(=O)N(CCCCN(CC)CC)C)N(C(=O)C=Cc1cc[nH]n1)C Cc1cc(=O)ccn1CC(=O)NC(C)C(C)(C)NC(=O)C(F)C(F)(F)F C1(CC(N2CC(NC(C3CCN(C(=O)OC)CC3)=O)C2)=O)CCN(OC)CC1 C1(OC)CC(NC(C2CC3C=CC2C3)=O)CN(C(c2cn(CCO)nc2C)=O)C1 c1(CCC(=O)NCC2CC2CNC(C2(CC(F)F)CC2)=O)ccc(F)c(F)c1 N1(C(CC(C)C(F)F)=O)CCC2(CCN(C(=O)CCC3CC3(Cl)Cl)CC2)C1 C1(CCNC(C2N(C(N)=O)CCC2)=O)CC2CCC(C1)N2c1cc(F)ncn1 CC(Cc1cnn(C)c1)C(=O)NC(CNC(C1(C#N)CCC1)=O)C1CC1 C(=O)(C(C)(C)C(F)(F)F)NC(C1CCN(C(C(COC)C)=O)CC1)C N1(C(CNC(CC)=O)=O)CCC2(CC(NC(=O)C(C)(C)N(C)C)CO2)C1 N1(C(C=C(C)C(C)C)=O)CCC(O)(CN(C(=O)C(C)CC#N)C)C1 c1(N2CCCC(CSC)C2)nc(N2CCC3CC3C2)nc2c1COC2 C=CCC(C)(CC)C(=O)NCc1nc(C(=O)NC2CCCCCC2O)co1 C1(n2cc(CCC(=O)Nc3ccsc3)nn2)CCCN(C(=O)CC2CCOC2)C1 N1(C(C2(CC=C)CCCCC2)=O)CC(NC(=O)CCCCCF)C(C2CC2)C1 C1(CCNC(C(CC)(C)OC)=O)CC(F)(F)CN1C(=O)C(COC)OC c1(CC)ccc(CCC(=O)NCC(CNC(C2C3CCN2CC3)=O)OC)cc1 N1(C(c2ccc(C(F)F)c(F)c2)=O)CC2CCC1C(Nc1ncnc(Cl)c1Br)C2 c1(C(Cc2cnc(NC(=O)CSc3ccc(C)cc3)s2)O)nc2ccccc2[nH]1 N1(C(=O)CC2CC2)CCN(C2CN(C(C3(F)CC=CC3)c3ccc(Cl)s3)C2)CC1 C(=O)(CC1COc2cc(OC)ccc21)NCC1(NC(C=CCOC)=O)CCOC1 N1(C(=O)NCC(c2ccc(Cl)cc2)C2CCC2)CCOC2CCCC12 c1(C(=O)NCC(CC)NC(=O)CNC(C)=O)oc(Br)nc1C c1(NC(C(=O)NCCc2c(OC)cccc2)=O)ccc2ccn(C(F)F)c2c1 c1(C(N(CCCNC(Cc2ncc(CC)[nH]2)=O)C(C)C)=O)ccc2ocnc2c1 C12(C(=O)NCCC3N(C(c4ccc(Cl)s4)=O)CCSC3)CCC(CC1)CO2 CN1C(=O)OCC1C(=O)NCC(CC(=O)N1CCCC1C1(C)CC1)N(C)C c1(OCC)c(CC(=O)NCCN(C(=O)CC2(O)CCCC2)CC)cccc1Cl C1(C(N(C)Cc2ccncc2F)=O)CCN(C(=O)Cn2ncn(C)c2=O)O1 N1(C(C(CC(CC)CC)F)=O)CCCC12CCCN(C(C1(CCO)CC1)=O)C2 c1(CN2CC(C(=O)O)CC(N(C)C)C2)c(F)cc(Br)c2c1OCO2 C(=O)(CC1=CCN(C)CC1)N(C)CC1CCC(NC(=O)COC(F)F)CC1 C1(CN(C)C(c2csc(-c3cccs3)n2)=O)C2CN(C(C3CCN(C)C3)=O)CC12 C1(C(=O)NC2CCCC(NC(c3ccncc3O)=O)C2)CC2CCC(C1)S2 c1(C(=O)NCCO)cccnc1N1CCCC(CCNc2ccccn2)C1 c1(Cc2nc(C3C(S(=O)(=O)C4CCC4)C3)on2)cccc2ccccc12 C1(CNC(C23CC(CC)(OC2)C3)=O)CC(C)(C)CN1C(c1[nH]nnc1C)=O C1(CC(N2C(CC(N)=O)CCC2)=O)CCCN(C(c2ccsn2)=O)C1 C(c1ccc(Cl)cc1)=CC.C12=CC=CC(O)=NC=C(C1=O)NCCNC2=O c1(C(C(=O)NCC(C)(C(C)C)NC(CC=CC)=O)C)ccc(F)cc1F N1(C(C=C(CC)C)=O)CC(NC(=O)C(C)=C2CCCC2)CC2(CC2)C1 C12(C(=O)NC3C(C(=O)OC)CC3)CC(C)(CN1C(=O)Cc1ccoc1)C2 c1(C(=O)NCC2(COCC)CC2)c(NC(C2CC=CCC2)=O)sc2ccccc12 c1(C(C)C)ccc2c(c1)C(NC(c1nc(CN(c3ccccc3)C)n[nH]1)=O)CC2 Cc1c(Br)ncc(F)c1CNC(C)C(c1ccccc1Cl)C c1(C(=O)NCC(CNC(C2ON=C(C)C2C)=O)O)c([N+](=O)[O-])cnn1C Cc1cccc2c(C(N3CCN(C(=O)CC4CCCCC4O)CC3C)=O)n[nH]c12 N1(C(C(C)OCCCC)=O)CC(O)(CCNC(=O)CCc2cc(Cl)cs2)C1 O(NC(=O)C1=CCN(C(C2CC=CC2)=O)C1)C(CC)CC N1(C(c2cnc(N)c(CO)c2)=O)CCOCC(F)(CNC(=O)CCSC(F)F)C1 C1(CNC(C(c2ccc(F)c(F)c2)C)=O)N(C(=O)CC2CSC2)CCC1(C)C c1(N2CCC(SC3CCC(=O)NC3C)C2)nc(NC(=O)OC)nc(=N)[nH]1 Cc1c(NC(=O)CCC(C)(C)NC(c2cc(Cl)n(C)n2)=O)cccc1C#N Cc1ccc(C)c(OCC(N2CC3(CCC3NC(C3CCCC(=O)O3)=O)C2)=O)c1 N1(C(c2cc(C(CC)C)no2)=O)CC(NC(c2nccnc2N)=O)C2(CC2)C1 C1(CNC(COCCC=C)=O)CC(NC(c2cc(C)ccc2F)=O)C12CCC2 N1(C(Cc2c(C)scc2)=O)CCOC(CNC(=O)Cc2ccc(O)cc2)C1 c1cc(F)c(F)cc1F.c1(C(C2(C)CC2)N)nnnn1CCC(c1ccsc1)C c1(C(=O)NC2CCCC(NC(C3(O)CC(F)(F)C3)=O)C2)cnc2cccnc2c1 c1(C(=O)NCC2(CNC(=O)CC(F)(F)F)CC2)cc2cc(Br)ccc2[nH]1 C12(NC(=O)CCF)CCCN(C(=O)CCN3CCOCC3)CC1C2 C1(NC(C(c2c(CC)cccc2)(F)F)=O)CCCCCC1NC(c1cnc[nH]1)=O N1(C(C(C)c2ccsc2)=O)Cc2ccccc2C1CNC(=O)C(F)OC(F)(F)F CCC(C(=O)N1CCC(CN(C(c2ccnc(CO)c2)=O)CC)CC1)C(C)C C1(OC)CN(C(=O)C(n2ccc(C)n2)C)CC1NC(=O)C=Cc1nccs1 c1(C(=O)NC(CCOC)C(=O)N(C)Cc2nc(C)no2)ccc(C)c(O)n1 C1(C(=O)NC2CC(NC(CSc3c(C)n[nH]c3C)=O)C2)CC2(C1)CC(C)(C)C2 c1(C(N(C2CCC(C)C2)CCOC)=O)cc(OC)c(F)cc1OC c1(C(=O)NCC(CNC(C2C(C=C)C2)=O)(C)O)n[nH]c2ccc(F)cc12 Cc1nc(NC2CC3CC(C2)N(C(=O)CCC2CCCCO2)C3)c(C)c(O)n1 N1(C(c2ccc(OC)cc2)=O)CC(=O)NC2CN(C(c3ns[nH]c3=O)=O)CCC12 c1(C(=O)NC2CCCN(C(c3c(C)cn(C)n3)=O)C2)c(C)ccc2nonc12 Cc1ccc(F)c(C(N2CC(C(N3CCCC(CCO)C3)=O)OC(C)C2)=O)c1 N#Cc1cc(F)ccc1C(N1CCC=C(C(=O)Nc2cccc3nsnc23)C1)=O C=CC1CCCN(Cc2coc(-c3ccc(Br)cc3)n2)C1 Cc1ccc(C(=O)NNC(=O)C2(c3ccccc3)CCN(C)C2)cc1Cl C1(C(=O)NCCN(C(C(n2cc(C)nc2)(C)C)=O)C2CC2)(NC(N)=O)CCCCC1 N1(C(C)=O)CCC2(CC1)CN(C(c1cccc3c1OCO3)=O)C2C(C)C C(C(C)(C)C1=CCCC1)NC(c1c(C)cn(C)n1)c1nnnn1CC1CC1 C1(N(C(C(C)N(C(C)=O)C)=O)C)CCC(CNC(C2(C)CC=CCC2)=O)CC1 OC1CC2(CCN(Cc3cccc(-c4cccc(Cn5ccnc5)c4)c3)CC2)C1 c1(CNC(C2CCC(C)O2)=O)ccc(CNC(=O)CC2CC2(C)C)cc1 c1(CCC)nnsc1C(=O)NCCC(C)NC(=O)Cn1nnc(C)n1 CN1CCN(C(=O)CC23COC(CF)(C2)C3)C(CNC(c2cnc(N)c(Cl)c2)=O)C1 CCC(C(=O)NC1(C)CC(C(=O)NC2(c3ccccc3Cl)CC2)C1)C(C)O C1(OCC)CCC(C(=O)NCC2(OC)CN(C(=O)CC3CCCCN3C)C2)CC1 C12(C(=O)NCC(C)NC(c3ccnc(C(F)(F)F)n3)=O)COCC(C1)C2 c1(NC(C23CC(C(=O)Nc4ncc(F)c(Cl)n4)(C2)C3)=O)c[nH]c2c(Cl)cccc12 C(=O)(C1=CCCCCC1)N1CCC(O)(C(C)NC(C=CCCC)=O)C1 c1(CSCC(C)O)nnc2ccc(C(F)(F)F)cn12 c1(CC)ccc(CN(C(c2ccncc2)C(=O)NCCCOC)C)cc1C CCCC(C)CC(C)(c1nnnn1C(C)(C)C)Nc1ccc(-c2cnco2)cc1 Cc1cc(C(=O)NCC(C2CCCCC2)NC(c2coc(CC3CC3)n2)=O)c[nH]1 CC1CN(C(=O)CC2CCCCN2C(=O)OC(C)(C)C)CCO1 c1(C(N2CCC(N(C(=O)C(C)n3cccn3)CC)C2)=O)cc(F)c(F)c(O)c1F c1(C(N2CC(CC=C)(NC(=O)CCn3cc(Cl)cn3)C2)=O)cc(C)cnc1Cl C1(NC(C(C(CC)C)c2ccccc2)=O)CCc2ccnn2C1 C12(CNC(C(C(C)(C)O)F)=O)CC(CCO1)N(C(c1ccc(CO)cn1)=O)C2 c1(C(N2CC(OCCNC(CN(C3CCC3)C)=O)C2)=O)ccc(F)c(Cl)c1N C(C1CCc2ncnn21)N1CC(NC(C2(c3cc(C)no3)CCCC2)=O)C1 N1(C(C2(CC3CC3)CC2)=O)CC(NC(C2(CF)CCC2)=O)C(c2ccccc2)C1 CC(C)C(F)(CNC(c1cc(Cl)cs1)=O)C(=O)N1OC2CCC1C2 c1(C(=O)NC2CCC(C(=O)NC3C(C)(COC)CCC3)C2)ncc2ccccn12 CC(C)CC(C)(CNC(=O)COC1CC(F)(F)C1)NC(=O)CCC(=O)N(C)C C1(CCC(=O)NC2C3CN(C(C(CSC)C)=O)CC2C3)CCc2ccccc2C1 O=C(C(F)(F)C(O)C1CC1)NCC1C2CN(c3ccc(Cl)nn3)CC12 Cc1cc(F)c(C#N)cc1NC(C1CCCC1NC(c1ccc(CO)o1)=O)=O CCC(C(=O)NCCCF)OC.C12(CCC1)C(=O)NCCOC2=O.C1CO1 C1(C(N2CCN(C(C(n3cc(Cl)cn3)C)=O)C(C)C2)=O)(CF)CCC(F)(F)CC1 Cc1ccc(C(N2CC(O)(C(F)C(=O)NC3CCC(=O)NC3)C2)=O)c(C)c1 C1(CNC(C(C)SC)=O)CC2(CC2)CN1C(c1cnc(C(C)(C)C)nc1C)=O C1(C)(C(=O)NCC(N(C(CCCOCC)=O)C)C2CC2)CCN(C)C1 c1(C(=O)NC2(CCOC)CCN(C(CC=CC=C)=O)C2)cc2n(c1)CCSC2 Cc1c(C(=O)NC2CN(C(=O)C=CCOC(C)(C)C)C2)cnn1-c1nccs1 c1(C(=O)NCCC(C)NC(=O)C(c2ccc(Cl)nc2)(F)F)ccc(N)c(F)c1F CC(C)(CC(=O)NC1CC(NC(c2coc3c(Br)cccc23)=O)C1)C(F)(F)F c1(C(=O)NCC(CN(C(c2cn(CC(CC)O)nn2)=O)C)O)cc(=O)n(C)o1 CC1CCC(NC(=O)C(N2CCOCC2=O)C)CN1C(=O)Cc1cc[nH]n1 C(=O)(CCC1=CCCCC1)NCC(C)(F)CNC(C1(CO)CCCO1)=O C=CCCC(O)CN(C(=O)CN(C)C(c1nonc1CC)=O)C c1(C(N2C(CO)CC(NC(C3CC34CCOCC4)=O)C2)=O)ncc(Cl)cc1F CC1NC(=O)CCC1CNC(=O)Nc1ncnc(C(C)(C)C)n1 CC(C)CC(F)(F)C(=O)NCC1(C)CCCN(C(=O)CC2CCCC2C)C1 CCCCS(=O)(=O)CC(=O)NCCCCCCNC(=O)C(CO)N(C)C c1(CC)ccc(C(=O)N(C)CC2COCCN2C(c2oncc2C)=O)nc1 N1(C(C)=O)CCC(NC(=O)C(O)Cc2ccccc2)c2ccccc21 CC(C)S(=O)(=O)C(C)C(=O)NCC1(CC#N)CCN(C(C2(C)CC2)=O)C1 c1(C(=O)NCC(CNC(CC2C(C)=NNC2=O)=O)(C)F)nc[nH]c2nccc1-2 c1(CN2CCOCC(C(=O)NCCOC(C)(C)C)C2)c[nH]c2ncc(Cl)cc12 N1(Cc2cc3cc(C(=O)OC)[nH]c3s2)CCSc2ccc(C)cc21 C1(C(=O)OCC)CCN(C(=O)CC2(OC)CN(C(=O)CCc3cccs3)C2)C1 C1(NC(CCCCC)=O)CC12CCN(C(C1CCC(=O)N1CCC)=O)CC2 C1(C(N2CC(CC=C)(NC(=O)CN3CCC3C)C2)=O)Cn2c(C)nnc2CN1C C(CN=c1[nH]c2c(c(=NCCC=CBr)[nH]1)CC(C)CC2)c1cc(C)sc1C c1(C(N2CC3C(CNC(C=C4CCN(C)CC4)=O)(C3)C2)=O)cc2ccccn2c1 N1(C(CCCOC)=O)CCC(C)C(NC(=O)COCC2CC2)C1C C(=O)(C1=NNC(=O)C1)N1C(CC(N2CC(C)(CCO)C2)=O)CCCC1 c1(C(C)C)noc(CCC(=O)NC(CNC(C2COCCO2)=O)CO)n1 CC(C)(O)C(F)C(=O)NC1CCCC1NC(=O)Cn1cc(F)ccc1=O Nc1c(C(=O)NC2COCCC2NC(=O)Cc2ccnnc2O)cnn1CCO CC1OC(C)C(C(N2CCOCC(NC(C3(S(C)(=O)=O)CC3)=O)C2)=O)C1C N1(C(C=CCC)=O)CCC2(CC1)CN(C(C1(C)CCN(C(C)=O)C1)=O)CCO2 c1(NCC(CC)NC(=O)OC(C)(C)C)nccc(=NCC2(O)CCC2)[nH]1 c1(OC)nc(C)ccc1C(=O)NCC1CCCN1C(=O)Cc1ccc(C)nc1 c1(CN(c2ccccc2NC(c2sc(Br)nc2Cl)=O)C)ccc2c(c1)OCO2 Cc1cncc(C(=O)NC(C(=O)NCCCCCCC2CC2)c2cccs2)n1 c1(C(=O)NC2(CNC(c3cccc(SCCC)c3)=O)CCC2)ccc(N)cc1F c1(OC)cc(F)ccc1C(=O)NC1CN(C(c2cc(C(F)F)no2)=O)CC12CC2 N1(C(c2n(C)nnc2Br)=O)CCCN(C(=O)Cc2cccc(F)c2)CCC1 C1(C(=O)NOCc2cnn(C)c2)(OCC(C)(C2CC2)OC)CC(F)(F)C1 C=Cc1cnn(C)c1C(=O)NCCC(O)CNC(c1ccc(C)cn1)=O C1(c2cccnc2)(C(=O)NCC2C(NC(=O)CCOC3CCOC3)C2)CCCC1 C(=O)(C(C)CCC(C)(C)C)NCC(CC(=O)NCC(F)(F)CO)OC N1(C(c2sc(C)c([N+](=O)[O-])c2)=O)CC(C)CN(C(c2cscc2F)=O)CC1C C(c1cccc(-c2cc(F)cnc2F)n1)=CO N1(C(CCCCC(C)=O)=O)CC(C2CCCN(C(=O)Cc3cnsc3)C2)C1 N1(C(CNC(C(n2c(C)ccn2)C)=O)(C)C)CCN(C(=O)C(C)CN(C)C)CC1 N1(C(C(CC=C)(C)C)=O)CCC(C2(NC(C3(Br)CC3(F)F)=O)CC2)CC1 N1(CC2OCCC2)CC2CCC1CN2CC1CC2CC2C1 C(c1ccc(F)cc1)=C(C)C(=O)NC1C=CCN(C(=O)Cc2ccc(Cl)cc2)C1 CC1=C(C)CC(C(N2CCCCC2CC(=O)NCC(=O)OC(C)C)=O)CC1 C1(CC(=O)NCCCN(C(=O)Cc2csc(C)c2)CCC)CCCC(C)(C)C1 Cc1coc(C2CC2)c1C(=O)ON(c1coc(Br)n1)CCC1CCCC1 Cc1[nH]nc(Cl)c1C(=O)NCC1(F)CC(NC(=O)CC2(C)CCCO2)C1 C1(C(=O)OCc2ccccc2N2CCOCC2)CCC(C2CCCO2)O1 C1(O)CCCN(C)C1=O.C1(CNC(C(C)C)=O)CCCCN1CCO C(CC(C(C)(C)C)NC(=O)Cn1ncc(O)nc1=O)N(C)C(C1CC1(C)C)=O CC(CC(=O)N1CCCC1CN=[N+]=[N-])C(C)(C)NC(=O)CN(C)C c1(OC)ccc2c(c1)CC(C(=O)NC1CC3CC1CN(C(c1ccco1)=O)C3)O2 c1(C(=O)NC2CCCN(C(c3cc(O)ncn3)=O)C2)c(Br)nc2n1CCC2 C1(NC(c2ccnn2CF)=O)CN(C(=O)CN2CC=CC2)CC1CC1CC1 C(C(CC(C)C)C(=O)NCC1CC(NC(=O)CCCF)C1)OC C1(CNC(C2CC(C(=O)OC(C)(C)C)C2)=O)CC(O)CN1C(C1CC1(F)F)=O O(N(C(=O)C1COCC1NC(C1C=CC1C(=O)OC)=O)C(C)C)CC C(N=c1nc(N2CCC(c3nncn3C)C2)c2c([nH]1)COC2)c1snc(C)n1 Cc1ncsc1CCC(=O)N(N(C)C)Cc1cn(CC(COC(C)C)(C)C)nn1 C1(C(C(=O)NC(C(=O)NCCC2(CO)CCC2)C2CCOC2)=O)CCCCC1 c1(C(N(C2CCCC2NC(C2(c3cccc(Cl)c3)CC2)=O)C)=O)ccc(=N)[nH]c1 C1(NC(c2n(CC)cc(Cl)c2)=O)COCCN(c2nccc(C#N)n2)C1 CC(C)C(C(=O)N(C)CCc1ncon1)C(C)NC(C1CC2CC(=O)C1O2)=O N1(C(CC=CCC)=O)CCC(O)(CNC(c2coc(N(C)C)n2)=O)C1 CC1(C)COCCC1C(=O)NC1CC(CCC(=O)NC(c2ncc[nH]2)(C)C)C1 c1(OC)c(-c2cn(CC3CC(F)(F)CN3Cc3ccccc3)nn2)cccc1F C(=O)(C(F)CCC(C)C)NC1(CNC(c2cc(CC)c(Cl)cc2)=O)CC(OC)C1 N1(C(C)(C)C)CCN(C(c2n[nH]cc2NC(C2CNC(=O)C2)=O)=O)CC1 C(=O)(C(C)(C)CCC#N)NC1(C(N2CCC(CC(C)C)C2)=O)CC(O)C1 c1(CC(=O)NCCc2n(CCC)cnn2)ccc(OC2CCCCO2)cc1Br c1(OC)cc(NC(C2COCCN2C(c2cc(C)ccc2F)=O)=O)nc(Cl)c1 C1(C(=O)NC2(CC=C)CN(C(C3CC(CF)C3)=O)C2)CCCNC1=O N1(C(c2nnn(C(C)(C)C)n2)C(=O)NC2(C)CC2)CCC(C2CC2(F)F)C1 C(CCC[Si](C)(C)C)NC(c1c(C)cc(C(F)(F)F)s1)C c1(C(=O)Nc2ccc3nc(C(F)F)oc3c2)cc(O)nc2cccnc12 N(C1CCc2cc(F)cc(Br)c21)C(C1(N)C(C)CCC1)=O c1(C(N2CCC(NC(C3N(C(=O)OCC)CSC3)=O)C2)=O)nccc2n[nH]cc12 n1(CC(C)C(N2CCCN(C(C34CC(C)(C3)C4)=O)CC2C)=O)ccc2ccccc12 c1(CNC(=O)NC(CC=C)CO)cc(C)ccc1C(F)(F)F C(=O)(CCC(=O)NC1(CNC(C2CCC(F)C2)=O)CCC1)N(CC)CC C(c1ccc(O)cc1)=CC(=O)N(CCCCNC(C(=O)NCCOC)=O)C1CC1 C1(C(=O)NCC=CCNC(=O)C(O)CN2CCCC2)OCCOC12CCC2 C1(C(N)=O)CCC(NC(=O)Cn2cc(CCc3ccccn3)nn2)C1 CCCCCC(=O)NC1CCOC(CNC(=O)CCc2cc(C)[nH]n2)C1 c1(CN(C(=O)NC2C(c3n(C)ccn3)C2)C2CC2)ccc(-n2cncn2)cn1 C1(C(N(CC(C)SC)C)=O)CCN(C(c2cccnc2S)=O)C1C N1(C(=O)CO)CCN(C(=O)C(c2ccccc2)NCc2ccc(Cl)cc2)CC1 c1(C(=O)NCC2OCCCN(C(c3c(SC)ccs3)=O)C2)c(C)ncn(C)c1=O c1(C(N2CCC(CNC(C(C(C)C)O)=O)C2(C)C)=O)ccc2cccc(O)c2c1 C1(C(=O)OC)CN=C2N=C(CN3CC(C4CCC(C(N)=O)O4)C3)NN2C1 CC1CN(C(C2COCCO2)=O)CC1CNC(=O)CSCC#N c1(C(N(C2CCN(C(=O)CC#N)C2)CCC)=O)ccn2cc(C)nc2c1 N1(C(c2n(CC)nnc2)=O)CC2(NC(=O)C(C)CN(C)C)CCC1CC2 C1(CCNC(C(c2cccc(C)n2)(F)F)=O)CCN(C(=O)CCF)C(C)C1 C1(C(=O)NCC(C)NC(=O)C(C)(C)O)CCCC1(F)F Cc1c(C(=O)N(C)CC2CCCN2C(C2(C)CC(O)CN2C)=O)cc(O)cc1N c1(CC)c(C(=O)NC2CC(O)(CNC(C3(C)CC3(Cl)Cl)=O)C2)cnn1CC(C)C c1(-c2cn(CCC(=O)NCC3(C)N=C(C)SC3)nn2)ccc(C#N)cc1 CC(C)(C(=O)N1CCCC1Cc1cn(C2(C3CCCNC3=O)CC2)nn1)C(F)(F)F CC(CC(=O)NCC(O)C(N)=O)NC(=O)C=C1CCC1 c1(C(=O)NCCN(C(C)C)C(c2ccnc(C(F)(F)F)c2)=O)csc2nccn12 C(=O)(CCCCCO)N1C(CN(C)C(C2(C(F)(F)F)CCC2)=O)CCC1 c1(C(=O)NCCN(C(CCC2CCC(C)O2)=O)C2CCCC2)nccc(Cl)c1O C(=O)(C(O)(C(F)(F)F)C1CC1)NCCCN(C(C1(OCC)CCC1)=O)CC N1(C(c2c(Cl)cn(C)n2)=O)CC(NC(C2CC3(CCC3O)C2)=O)CC12CCC2 c1(C(C)=O)cnc(N(C(=O)NCC2CCC(C)(C)O2)CC2CCCO2)c(C)c1 C1(CCC(C)C)C(=O)N=C2C=C(C)N1N2.Cc1c(CN)cccc1F N1(C(c2cc(OC)ns2)=O)Cc2ccccc2C(NC(c2c(C)n[nH]c2C)=O)C1 c1(CC(=O)OCC)noc(C2CN(C(=O)C#CCNC(C3CCC4CC34)=O)C2)n1 C1(n2c(-c3c(C)nc(Cn4cccn4)s3)nc(C(C)C)n2)CCS(=O)(=O)CC1 C1(CC#C)(C(=O)NCCN(C)Cc2csc(-c3ccc(C)cc3)n2)CCCCO1 c1(C2C(CNC(c3nc4cccc(Br)c4[nH]3)C)C2)ccc2c(c1)OCCO2 CCCC(C(=O)NCC(C)(C(C)C)NC(=O)CCOC)c1ccccc1 C(=O)(CC(C)CC(C)(C)C)N1CCC(CC=C)(NC(C2CC(F)(CO)C2)=O)CC1 Cn1ncc(NC(=O)Cc2cc(Cl)c(Cl)s2)c1-c1cn(CCC(C)(C)C)nn1 Cc1ccc(C2CCN(C(C3CCOCC3)C(=O)NC3COC3)C2)c(C)c1 N1(C(c2c(C)ncnc2)=O)CCC2(NC(c3cn4c(n3)CCC4)=O)CC2C1 N1(C(CCCC=CCCC)=O)CC2(CCN(C(=O)CCc3ccc(SC)cc3I)CC2)C1 N1(C(c2c(OCC#C)cc(Br)cc2)=O)CCn2nc(COC)cc2C1 c1(C(=O)NC2(CC)CCCN(C(C3(O)COC3)=O)C2)cnc2ccc(C)cn12 N1(C(c2ccc(C(C)(C)C)cn2)=O)CCC2C(C1)CN2C(c1ccncn1)=O Cc1cc(C2CC2)ncc1C(N1CCCC1C(C)NC(=O)CC1(C)CC1(F)F)=O C1(NC(c2c(OCC)oc(C)n2)=O)CC2CC1CN(C(C13C(=O)C4CC1C3C4)=O)C2 C1(NC(C2C(C)C2)=O)CCN(C(=O)CCS(=O)(=O)N2CCOCC2)CC12CCC2 CC1CNC(C)(C)CN1Cc1ccc(Br)c(Br)c1 C1(NC(C2C(C(=O)OC)C2)=O)CCN(C(c2ccc(F)cc2C)=O)CC1O CCCC(CCC)CCCC(=O)N(CCC(C)NC(=O)CC1CC(OC)C1)C C1(NC(C2(NC(C3CCCCC3(F)F)=O)CSC2)=O)C2CCCCCC12 CCC(CC)C(C)C(=O)N1CCC(C2CC2)(NC(=O)COc2ccccc2C)C1 C1(C(=O)NCCCNC(c2cn(CC(=O)N(C)C)nn2)=O)CC(S(C)(=O)=O)C1 C1(NC(c2c(CC)nc[nH]2)=O)COC2CN(C(=O)C3=CCCCO3)CC12 C12(NC(c3cccc(OC)c3F)=O)CCCN(C(c3scnc3Cl)=O)CC1C2 CN1CCOCC1C(N1CCC(C)(CNC(=O)CSC(F)F)C1)=O CC1CC(CC(N2CCC(CC(N)=O)CC2)=O)CN1C(=O)CN1CCCCC1=O CCC(C)C(O)CNC(c1coc(CNC(c2ccc(C#N)o2)=O)n1)=O Cn1cc(C(=O)NCC(C)(F)CNC(C2SCCS2)=O)ncc1=O c1(CC)cccc(NC(=O)C(C)N(C(c2c[nH]c(=S)cn2)=O)C2CC2)c1F c1(OC)cc(OC)c(CN2CC(CNC(c3c(F)ccc(O)c3O)=O)C2)c(OC)c1 N1(C(CNC(c2c(C)cccc2)=O)=O)CCC2C1CCN2C(C1CCC1)=O CN1C(=O)CSC1=CC(=O)NCC1CCC(CNC(=O)CC2COCC2O)CC1 c1(C(=O)NC2C(CNC(c3ccoc3)=O)CCC2)nnn2c1C(=O)NCC2 c1(C(=O)NCC2(O)CN(C(CC3CCCC(C)C3)=O)C2)cnc2c(c1)COCC2 c1(C(C)O)ccc(C(=O)NCCCC(CO)NC(=O)Cc2ccc(O)nc2)cc1 C(=O)(C(F)CC(C)(C)NC(C12C(=O)C3CC1C2C3)=O)NC1CC(C)(C)OC1 c1(NC(=O)NCC(CC)CO)cc(N2CCN(C(C)=O)CC2)ccc1F c1(C(=O)NCCC(C)NC(=O)C(C)(C)Cc2cnn[nH]2)c[nH]c2cccc(F)c12 N1(C(CCc2onc(COC)n2)=O)CCC(C)OC(C)C1 c1(C(=O)NCC2OCCC(NC(C(C=C=C)C)=O)C2)ccc2c(O)ncnc2c1 CC1CCN(C(C2CC(C)CC(C)C2)=O)CC1CNC(=O)CCNS(C)(=O)=O N1(C(C(C=CC)O)=O)CC(NC(=O)CCSCc2ccccc2)C(C)(C)C1 C1(NC(Cc2cccc(OC)c2)=O)C2CC3CN(C(=O)C=CBr)C1C3C2 N1(C(=O)CSc2cccc[n+]2[O-])CCC2CCN(C(=O)CC3CCCOC3)C2C1 c1(OC)cnnc(C(=O)NC2CCN(CC(=O)NCc3ccc(C)cc3)C2)c1 C(C(O)C(C)(C)C)NC(C(C)(C1CCC1)NC(C(C1CCC1)OC)=O)=O c1(C(C(=O)NC(C(C)NC(C2CC(CC)(CC)C2)=O)CO)O)cn(C)nc1C C1(O)(CN(C(C(C)NC(=O)NC)=O)C)CN(C(=O)C(O)Cn2cncn2)C1 C1(C)(C(=O)NCCN(CC(C)O)C(c2ccc(C(C)(F)F)cc2)=O)COCCO1 C1(C(CNC(C(C)=CC)=O)(C)C)CCCN1C(=O)C(CC)NC(c1ccco1)=O C(C)(CC(=O)NCCCOCCNC(=O)CCCN1CCCC1)SC N1(C(c2nccc(OC)c2C)C(=O)NCCC)CCC2(CC1)C(=O)NCCN2C Cc1ccc(C=CCC(=O)NCCCCC(C)NC(=O)C=Cc2cscn2)cc1 N1(C(c2csc(C(C)(C)C)n2)C(=O)NC)CCc2cccc(C(F)(F)F)c2C1 c1(C(=O)NCC2(F)CN(C(CC)=O)C2)ccc(C)c(S(=O)(=O)CCO)c1 C1(C(=O)NCCN(C(c2cc(S(N)(=O)=O)cs2)=O)CC)CNC(=O)CC12CCC2 Cc1cc(C(N2CCN(C(=O)C(C)NC(C)(C)C)CC2C2CC2)=O)ccc1Cl C(=O)(CC1OCCc2ccccc21)N1CCC(C(C)NC(C(C)OC)=O)C1 Cn1nnc2ccc(C(N3CCC4CCC(C3)N4C(c3cnc[nH]3)=O)=O)nc12 C1(C(N(C2CC(NC(CCCNC(C)=O)=O)C2)C)=O)CN2CCC1CC2 C12(C(N(C3CC(CNC(=O)C(O)Cc4ccccn4)C3)C)=O)CCN(CC1)CC2 N1(C(C(C)OCCC=C)=O)CC2CC(NC(=O)C=CSCc3ccco3)C(C2)C1 c1(C(N2C(CNC(C(CC#C)(C)C)=O)CCC2)=O)noc2c1CN(CC)CC2 C1(NC(COC2(C)CCC2)=O)CCCN(C(=O)CCCc2ccc(Cl)cc2)CC1F c1(C(C)NC(C(C)SC)=O)ccc(CNC(C2CC3CCC3C2)=O)cc1 Cc1cccc(C(=O)NC(C2CCCC2)CNC(=O)CC2CCC(=O)C2)c1C C1CC(C(C)C)N1C(C(CC)n1cccn1)=O.C1(OCC)CCCOC1.C1(=O)CO1 c1(C(=O)NC(CC)(C)CNC(c2nn(C)cc2C)=O)ccc(N)cc1S(N)(=O)=O c1(NC(C2CCC(CNC(=O)NCCCl)O2)=O)ccccc1F.C12CCN1C2=O C12(NC(C(CC#C)C)=O)CCC(CNC(c3ccc(C(C)C)cc3)=O)(CC1)OC2 c1(C(=O)NC2CCN(C(CS(=O)(=O)NC)=O)C23CC3)cnc2cnn(C)c2c1 N1(C(C2CCC(C)O2)=O)CCN(C(=O)C(O)C2CC2)CC1C C(=O)(CCCCCC#N)NCC(CC)N(C(=O)C(c1ccc(C)cc1)F)C c1(C(N(CCNC(CC(C)C2CC2)=O)C)=O)ccc(S(C)(=O)=O)cc1 c1(C(=O)NCCC2(O)CCN(C(C3(C#N)CC=CC3)=O)C2)nc2ccccc2[nH]1 C(=O)(C1Cc2ccc(Cl)cc21)NC1CC(C)(C)N(C(c2cnc3n2CCS3)=O)C1 C1(CC(=O)N(CCCCCNC(c2c(C(C)C)con2)=O)C)COCC1(C)C c1(CN2CC(NC(c3c(OC)ccs3)=O)C(F)(F)C2)cc(Cl)c(Cl)nc1Cl C1(CC)C(=O)NCCN1C(C1CC(O)CN1C(=O)C1=CCCCO1)=O Cc1nc(-c2ccccc2)sc1NC(c1cc(-c2ccco2)on1)=O c1(C(=O)NC2CCN(C(C(C)(C)C)=O)CC2F)ccc2c(Cl)ccnc2c1 CS(=O)(=O)c1ccsc1CN=c1cc(NCCOCCS(N)(=O)=O)nc[nH]1 Cc1ccc(CNc2csc(-c3ccccc3)c2)cc1C#N.N12CC=CC1C2=O Cc1nc2nc[nH]n2c(=O)c1CCC(=O)N1CC(NC(C2(C)CC3CC3C2)=O)C1 C1(CCCC)CN(C(=O)C(C(C)C)OCC)CCN1C(=O)CCc1scnc1C C1(C(=O)NC(CC)Cn2cncn2)(CF)CCN(C(=O)CCCCSC)C1 C(=O)(CC(C)C(F)F)N1C(COC)CC(CNC(C2(c3cccnc3)CC2)=O)C1 c1(C(=O)NCC2(C)CCCC2)ncccc1NCc1cccnc1C(F)(F)F N1(Cn2ncc(CC)c2)CC(C(=O)OC)OC(C)C1 Cc1ccc(S(=O)(=O)NC2(c3ccc(F)cc3)CCCCC2)c(C)c1 O=NN1CCCC1C(=O)NCC1CC(F)(CNC(c2ccncn2)=O)C1 c1(C(=O)NCC2(O)CCN(C(COCCC=C)=O)C2)c(C)sc2ccc(F)cc12 N1(C(C2C(CCC)CCC2)=O)CCCC2CN(C(=O)CC34CC(C3)C4)CC12 C1(NC(C(Cc2ccco2)NC(C(C=C=C)C)=O)=O)CC2CCC(C1)N2C Cc1cccc(CC(=O)NCC(C)(O)CNC(=O)Cc2ccn(C(C)C)n2)c1Cl n1(CC(=O)N(C)CC2CCCN2C(=O)CCc2ncco2)nnc2ccccc12 N1(C(C2N=C(C)SC2)=O)CCC(CNC(c2n[nH]cc2Cl)=O)C(F)(F)CC1 C=CC(C)(O)C(=O)NCCN(CCC)C(C1CC(C)CCO1)=O c1(C(=O)NC(C)CCNC(=O)CN(C)C(N)=O)cn(C)nc1-c1ccnn1C c1(NC(C2C3C(=O)OCC23Br)=O)cc2c(s1)COCC2 C(=O)(C(C)S(N)(=O)=O)NC1(CF)CCN(C(C2CC(C(=O)OC)C2)=O)C1 c1(C(=O)NC2(CC(N3CC(C(=O)OC)(SC)C3)=O)CCC2)cc(C)n(C(C)C)n1 N1(C(C(=O)Nc2c(OC)ncnc2C)C)CC2CCCC2(N)C1 N1(CCC(N2C(CN(C)C)CCC2)=O)C(=O)C2CC=CCC2C1=O c1(C(=O)NC2CCN(C(C(C)c3cc[nH]n3)=O)CC2)ccnc2[nH]ncc12 c1(C(C(=O)NC(CNC(C(C)SCC)=O)C2CC2)(F)F)ccc(F)cc1F c1(CC)c(C(=O)NC(C)CNC(=O)C2=CC3CCC2C3)sc2ccccc12 c1(C(N2CCCC(CCNC(C3COCCO3)=O)CC2)=O)ccc2cccnn12 C1(CNC(c2cnc(C(C)OC)s2)=O)COCCN(C(=O)CN2CSCC2=O)C1 Cc1sc(=O)n(CC(=O)NCCCN(C(C2C(C)(C)OC2(C)C)=O)C2CC2)c1C c1(-c2nc(CC(CC)C)nn2CCC2CC2)cccc(S(=O)(=O)CCO)c1 C1(C(=O)NC2(CC=C)CCN(C(C3(CC4CC4)CCC3)=O)C2)COCCC1(F)F C1(C(N)=O)(CNC(CC=C)=O)CN(C(=O)C(n2ccc(C(=O)OC)n2)C#N)C1 C1(CC(=O)NCc2n(C(C)C)cnc2)N(C(=O)C(C)C2CCOC2)CCC1(C)C N1(C(=O)CC(C2CC2)C2CC2)CCN(C2CCCN(C(C3CC(O)C3)=O)C2)C(=O)C1 CCCCC(O)C(C)C(=O)NCC1CCN(C(c2ccc(COC)o2)=O)C(C)C1 N1(C(c2c(C)n(C)nn2)=O)CCC2(CCCCC2NC(=O)Cn2cc(Cl)cn2)C1 N1(C(C2CC(OC)C2)=O)CCC(F)(CNC(c2nc(=N)cc[nH]2)=O)C1 C(CC(C)C(=O)NCc1cncc(C(=O)NCC2(F)CN(C)C2)c1)=CCC c1(N(C)Cc2nncs2)nc2cc[nH]c2c(=NC2CC(c3ccccc3)C2)[nH]1 S(=O)(=O)(c1cc(C)cnc1NCCOC(F)F)NCC(c1ccc(OC)cc1)O S(=O)(=O)(c1cnc2ccsc2c1)N(C(c1ccc(SC)cc1)=O)C(C)C c1(C(=O)NC2CN(C(CC3C(C)(C)CCO3)=O)C2)ccc(C#N)c(C(F)(F)F)c1 CC1CN(C(=O)C=Cc2cn(C)cn2)CC1(C)CNC(c1nonc1N)=O C12(C(N(c3c(C)cccc3)C)=O)C3C(=O)C4C5CC(C14)C2C35 N1(C(C2(OC)CCC2)=O)CC2CC1CN2C(c1cccc(Cl)c1Br)=O c1(OC(C)C)ncc(C(=O)OCC2C3CC=CCC23)cn1 N1(C(c2cc(C)c(C)[nH]2)=O)CC(C2CN(C(=O)C=Cc3cnc[nH]3)C2)C1 N1(C(C2(OC)CCS(=O)(=O)C2)=O)CCC2CC(NC(=O)C=CC(N)=O)CCC2C1 O=C(N=c1ccn(C2CN(N3CCn4cncc4C3)C2)[nH]1)C12CC(CO)(C1)C2 c1(C(N2CCCC(N(C(=O)C(C)C)CC)C2)=O)ncc(Br)cc1C N1(C(c2nccc(OC)c2)=O)CCN(C(=O)C(=Cc2ccccn2)C)CC1CO c1(C(=O)NCC(C)N(C(=O)C#CC2CC2)C)ccc2c(c1)OC(C)(C)OC2 CC1CN(C(c2ccnn2CCF)=O)CCCN1C(=O)CCC1CCC(=O)NC1 N1(C(C(C=C)(F)F)=O)CC(NC(=O)CCSC(F)(F)F)C2(CCC2)C1 Cc1cc(C)c(C(N2CC3(CNC(C4CCNC4=O)=O)CC2CO3)=O)c(C)c1 CS(=O)(=O)c1ccccc1CN1CC2C(Nc3ncnc4sc(Br)cc34)C2C1 C1(C(=O)NCCC(C)N(CCC)C)C=CCN(C(c2cnsc2)=O)C1 C(c1ccnc2ccccc12)=CC(=O)NC1CCCC(N(C)C(c2ccns2)=O)C1 C1(NC(=O)Cc2cnco2)CCOC(C2CCN(C(=O)C3=CCOC3)CC2)C1 c1(C(N2C(C)(CNC(C(CC)CO)=O)CCC2)=O)cccc2c1NC(=O)CO2 c1(C(N(C)CC2CCN(C(=O)COC(F)F)C2)=O)cccc(O)c1 C(=O)(CCC(=O)N1CC(N(C(=O)C(F)C(C)C)C)C(O)C1)N(CC)CC C1(NC(C2C3CN(C(C(CCC)NC(N)=O)=O)CC32)=O)CC2CC(O)C1C2 c1(COC)nc(C)c(C(=O)NCCC2CC(NC(=O)C(C3CCOCC3)F)C2)s1 C12(C(=O)NCC3CC(NC(CN=S(C)(C)=O)=O)C(O)C3)CCC(O)(CC1)CC2 C1(NC(c2cccc3nncn23)=O)CCC2CC1CN2C(c1csc(Cl)c1)=O c1(C(N2C(CC(=O)Nc3cc(C)c(Cl)cc3Cl)CCC2)=O)cccc2ncccc12 C#CC1CCCCN1C(=O)CCCCNC(c1cn(CC)nc1C)=O C(CCOCCO)(C(=O)N(C1CC=CC1)C)NC(CC(C)c1ccco1)=O c1(C(N(CCCN(C(C(C(CC)O)(F)F)=O)C)C)=O)cc(S(C)(=O)=O)ccc1C c1(OC(CC)C)ccc(O)cc1.c12ccc(cn1)CNC(=O)N(CCO)CC2 CCCC(C(=O)N1CCCC1(C)C(C)(C)C)NC(c1cc(CO)[nH]n1)=O C(c1ccccc1C#N)=CC(N1CCC(CCNC(c2c(C)nccc2)=O)C1)=O C1(CNC(c2cnc(Cl)[nH]2)=O)CC2(CCC2)CN1C(=O)CCc1nncnc1O N1(C(C2CN(C(C(C)=C(CC)C)=O)CC(C)C2)=O)CCC(F)(F)C(F)C1 C#Cc1ccc(C(=O)NC2CCC(NC(=O)C(C3CCCC3)OC)C2)cc1C N1(C(C(C)c2cccs2)=O)CCCC(NC(=O)CCOCC(F)F)CCC1 S(=O)(=O)(c1c[nH]ccc1=NC1CC2(CCCC2)C1)NCC(c1cccnc1)OC c1(C(=O)NCCN(C2CCCC2)C(=O)C=Cc2nccs2)c(F)cc(O)cc1F CC(C)C(C)C(C)CC(=O)N1CC(CNC(C23CC=CC(C2)OC3)=O)C1 c1(C(N2CCC(C(=O)NCCCN3CCOCC3)C2)=O)cc(F)ccc1[N+](=O)[O-] C1(C)(CNC(c2cnc(SC)s2)=O)CN(C(C23CCC(C2)OC3C)=O)CCO1 n1(C(CC)C)ncc(C(=O)NCC(C(C)(C)C)NC(c2coc(Cl)n2)=O)c1C N1(c2nc(Cl)c(C3CC3)cc2)CC=CCC2(CCOCC2)C1 C(=O)(CCC(=O)NCC(F)(F)Cn1cc(-c2cccc(F)n2)nn1)N(C(C)C)C c1(C(C(=O)NC2C(NC(c3ncc(F)cn3)=O)CCC2)O)ccc(Cl)c(F)c1 C1(C2CCN(C(=O)C=CCO)CC2)(CNC(c2cnc(C)n2C)=O)CCOCC1 N1(C(Cn2c(C)ccn2)=O)CC2(CNC(=O)CCC3CCCCC3)CC1CO2 C1(C2CCN(C(=O)CS(N)(=O)=O)CC2)(NC(c2c(C)n(CCO)cc2)=O)CCC1 C(CC(=O)NCC(=O)NCC(CO)NC(=O)CC1CC1(C)C)NC(C)=O c1(C(=O)NCCC(CNC(C2(CC)CCCC2)=O)O)ccc(O)c([N+](=O)[O-])c1 CCCC(C)(O)C(=O)NCc1ccc(C(=O)NC(c2ccccc2)CO)cn1 C1(C(=O)NC2C(C(=O)NCCSCCOC)CC2)(OC)CCCC1 c1(CCC)nc(C)c(C(=O)NCCN(CCC)C(c2sc(C(C)C)nc2C)=O)o1 C(C(C(=O)NCCCCC1CC1)NC(=O)COC)OCC.C1CCO1 N1(C(CC=C)=O)CCN(C(c2cc(-c3ccco3)[nH]n2)=O)C(CC2CC2)C1 N12CCC(CC1)C2=O.C(=O)(C(O)Cc1cnc[nH]1)NCCSC.CCCCN(C)C C1(C(NNC(C)=O)=O)CCN(CCNC(C(C)(C)C)=O)CC12CCC2 c1(C(=O)NCCC(C)NC(C=C(C)C)=O)cc(C(C)CC)no1 CC(CC#N)C(=O)NCC1CCCN(C(=O)C(C)(F)F)C1 C(=O)(C1=NOC(CNC(=O)CC(C)(C)C#N)C1)NCC(CC)(C)O N1(C(C2CCN(C(=O)NC)CC2)=O)CCCC2(CCN(C(=O)C(C)O)C2)C1 C12(NC(CC(C)(F)F)=O)CCCCCC1N(C(c1ccn3c1CCCC3)=O)CC2 C(=O)(C1(C)CCn2ccnc21)N1CC(CC(C)NC(c2oc(CC)c(C)c2)=O)C1 C1(C(N2C(C)CCC2)=O)CN(C(c2cn(C)ccc2=O)=O)CCN1C c1(C(N2C3C(NC(C4CC5CC5C4)=O)C(CC3)C2)=O)cccc2nn[nH]c12 S(=O)(=O)(c1c[nH]c(C(N2CC(NC(C3CC3OC)=O)CC(C)C2)=O)c1)NC c1(OC)cccc(F)c1NC(C1CCCN(C(c2oc(C)nc2C)=O)CC1)=O N1(C(c2nccc(N)c2)=O)CC2CCC(NC(=O)C(c3ccccc3)O)CC2C1 N1(C(C2C(OCC)CC2)=O)CCC(C2CC2)C1C(=O)NCc1ccc[n+]([O-])c1 N1(C(C(CCC#C)NC(c2cnsc2C)=O)=O)CCCC(C)(C)C1C n1(CCC)nnnc1C(c1occc1COC)NCCCc1cc(C)no1 CC(C)CCCCC(=O)NCC1CC1CNC(=O)COc1ccccc1O c1(C(N2CC(C(=O)NCC(C)(C3CC3)OC)C(C)C2)=O)cc2ncccc2[nH]1 C(=O)(C1=CCCCO1)N(C1CCCC1)CCCNC(C(n1cc(C)nc1)(C)C)=O c1(CN2CC(CC#N)N(C(=O)C=Cc3cccs3)CC2)ccc(F)c([N+](=O)[O-])c1 N1(C(=O)C(O)C(F)(F)F)CCN(C(=O)C(F)(F)c2ccncc2)CC(O)C1 N1(C(C(c2cccs2)SC)=O)CC2CC2(CNC(=O)CN2CCC(C)CC2)C1 C#Cc1cncc(C(=O)NC2(CNC(=O)C(O)(C(C)C)c3ccccc3)CC2)c1 C1(c2nnnn2C2(C)CC2)(NC(CSC)(C)C2CC2)CCCCC1CCCO c1(CC(=O)NCC(=O)NC(CC=C)CNC(=O)C=CC(F)(F)F)cccc(C)c1 c1(C(C(=O)NC2CCN(C(C3CCCCCC3)=O)C2)F)ccc(C(F)(F)F)cc1 N1(C(CCCC(=O)NCC)=O)CCC2CCCC12CNC(c1cc(C)ns1)=O C1(c2cn(CCOC)nn2)N(CC(=O)N(C(C)C)C(C)C)CC12CCOCC2 c1(CNc2nccc(N3CCCC(C)(C(=O)NC)C3)n2)ncccc1S(C)(=O)=O c1(C(=O)NC(CC(C)C)CNC(=O)CCCN(C)C)ccc2c(c1)C(=O)NCC2 N1(C(CC2CCC(=O)N2)=O)CC2CCCC(C1)N2C(c1cccc(=S)n1O)=O N1(C(c2ccnc(SC)n2)=O)CC2CCC1CN(C(=O)CCc1ccsc1)C2 N1(C(CCNC(=O)CO)=O)CCOC(c2cn(C3CCOCC3)nn2)CC1 Cc1cc(C#N)cc(CN(CCCCCCO)CC2CCC(C)(C)CC2)c1N c1(OC)ccc(C(=O)NCC2CC2NC(c2cccc(N)c2)=O)c(OC)c1Cl c1(C(=O)NC(C(C)NC(=O)C=CC2CCOC2)(C)C)cc(N)ccc1Br N1(C(CCNC(C2C(C)C2)=O)=O)CCCN(C(=O)C(O)c2cnc[nH]2)CC1 C1(CN2CC(C)(NC(c3cccc(CC)n3)C3CCCC3)C2)Cc2nccn2C1 c1(C(C(=O)NCCCN=[N+]=[N-])NC(=O)OC(C)(C)C)ccc(F)cc1 CC1C(C(=O)NCC(CC(N2CCC3(CC2)CSC3)=O)C2CCC2)=NOC1C c1(C(=O)NC(CNC(CCC(C)C)=O)C(C)(C)C)cc(C(F)(F)F)cc(N)c1 c1(C(C)NC(C(=O)N(C(CC)CO)CCc2ccccn2)=O)cc(Cl)ccc1Cl N1(C(C2(C)ON=C(C)C2)=O)CC2CN(C(c3cccn4nnnc34)=O)CC2(C)C1 C1(NC(=O)NC(C)C(=O)NCCF)CCC2CCCC1O2 c1(C(N2C3C(NC(CC(C)NC(N)=O)=O)CC(C3)C2)=O)cccc(C#CCO)c1 N1(C(c2cnn(CCC)c2C)=O)CCCC(C2CC2NC(=O)CO)C1 N1(C(CNS(CC)(=O)=O)=O)CC(C)(C)CC1CNC(=O)C(C(C)C)n1ccnc1 Cc1nc2ccc(C(N3CCN(C(=O)CC4(C)CC4)CCC3C)=O)cn2n1 C1(CN(C(c2cc(C)sn2)=O)C)COCCN1C(c1ccc(O)nc1)=O N1(C(COC)=O)CCC2(CC1)C(OC)CC2NC(C1CN(C2CCCC2)C1)=O N1(C(c2n(CC)ncc2Br)=O)CC2CC(C1)N(C(=O)C=CC(C)(C)SC)C2 O=C1N(CCc2ccc(OC(=O)OC(F)F)cc2)C(=O)C23CC(CN12)C3 N1(C(c2cn(C)nn2)=O)CC2(C1)CN(C(=O)C(CO)C(C)(C)C)CCO2 CCC(C)(CC)C(=O)NCC12CC(NC(c3ccn(C)c3)=O)(C1)C2 CC1(C)CC(C(=O)NOC2CC3CCC2C3)CN1C(=O)CCc1cccs1 c1(C(=O)N(C(C2N(C(C=CCN(CC)CC)=O)CCC2)(C)C)CC)ccc(C)nn1 C1(c2nnnn2C(C)(C)C)(NCc2cc(C)sc2C)CCC2CCC1C2 C1(NC(C(C)Cn2cccn2)=O)CC(F)(F)CC1NC(c1cnc(S)[nH]1)=O C(CC1CNC(=O)C2(CCCO2)C(=O)N1)OC.C1(N(C)C(C)=O)CCCC1.CO N1(C(C2CNC(=O)N2)=O)CC2(C1)CN(C(C1CCc3ccnn3C1)=O)CCO2 c1(SCC(=O)NCCCN(C(=O)CCc2ccsc2)CC)ccc(C)cc1F N1(C(c2ccc(C)nn2)=O)CC2CCC(N(C(=O)C(N)=O)C)C2C1 C(c1ccccn1)=C(C)C(=O)NC1CC1NC(c1cccc(SCC#N)c1)=O Cn1nc(C(=O)OC2CCCN(C(C3(C)CCOCC3)=O)C2=O)c(Br)c1Cl N1(C(CC(C)(C)F)=O)CC(NC(=O)CS(=O)(=O)N2CCCCC2)CC12CCC2 C1(CNC(c2cc(CNC(=O)CC3CSCCO3)oc2)=O)CC2(CCCO2)C1 CC1CN(C(=O)CC2(C)OCCO2)CC1CCNC(c1cnc(C(C)(C)C)o1)=O c1(-c2cc(C(=O)NCC(=O)NCc3ccncc3)sc2)ccnc2ccccc12 Cc1cc2ncc(CNC(N3CCC(CNC)C3)=O)cn2n1 C1(C(=O)NCCOCC#C)(NC(C2CC3CCCC3C2)=O)CCC(C)(C)C1 C1(NC(CCC(=O)NC)=O)CN(C(=O)CC2(O)CCN(C)CC2)CC12CCC2 c1(-c2cn(CC3C(CNC(CNS(C)(=O)=O)=O)C3(F)F)nn2)ccc(F)c(F)c1 N1(C(=O)NCCNc2cnc[nH]2)CCCCC1C1CCC1 C(=O)(CC(O)C(Cl)(Cl)Cl)NCCCN(C(C1(CC#C)CCOCC1)=O)C Cc1nc(-c2cccs2)sc1C(=O)NCCN(C(C1CCN(C)C1C)=O)C1CC1 N1(C(c2n(CC)ccc2)=O)CC2C(NC(C3CCN(C)C3=O)=O)C2C1 C(=O)(C(C(C)C)n1cncn1)NCC(C1N(C(c2cnc(C)s2)=O)CCC1)(C)C C(CCC(N)=O)(C(=O)N1CC2CC1C2NC(C1CCS(=O)(=O)C1)=O)N(C)C Cc1ccc2nc(NC3CCN(C(c4cnnn4C)=O)C(C)C3)sc2n1 CCCCCC(O)C(C)C(=O)NCC(C)(C)CNC(=O)Cc1c(C)ncnc1C c1(-c2cn(C(C)C(=O)N(C3(C(=O)O)CCC3)C)nn2)cc(Cl)c(Cl)cc1Cl C1(C(N2CC(C(C)C)OCC2)=O)CC2CCCCC2N1S(=O)(=O)c1ccccn1 Cn1cc(C(=O)NCC2CCN2C(=O)CC(O)C2CC2)c(O)nc1=O NS(=O)(=O)C1CCN(c2cc(NCc3nnc(Br)n3C3CC3)ncn2)C1 CCCC(CC)(c1nnnn1CCOC)NCc1ccsc1Cl N1(C(c2cc(C)n(CC)c2C)=O)CC(C2CN(C(=O)CC34CCC(CC3)C4)C2)C1 CN1CCCC(C(N2CC3C(CNC(=O)C=CCn4cncn4)C3C2)=O)C1 N1(C(CCn2ccc(C)n2)=O)CC(C)CN(C(c2csc(F)c2)=O)CC1C N1(C(c2n(CCCC)ncc2)=O)CC(NC(=O)Cc2cnnn2C)CCC1C N1(C(C2(CC=C)CC2)=O)CCC(CN(C(=O)CSCC(=C)C)C2CC2)CC1 N1(CC(=O)NC(C(C)C)CNC(C2CC2c2cncn2C)=O)CCCNC1=O Cc1ccc(NC(C2(NC(=O)C(C)CC#N)CC2)=O)c(C)n1 CCCCCCC(F)C(=O)NC1(C)CCCN(C(C2C3CCC4C(C3)CC24)=O)C1 N1(C(C(C(CC)C)O)=O)CC2CC(C(=O)NCCNC(=O)NC3CCCC3)CC2C1 c1(C(=O)Nc2n(C)nc(-c3ccccn3)c2)cccc([N+](=O)[O-])c1O O(NC(=O)C(C1(O)CCC1)NC(=O)C(C1CCCCC1)O)C(C(C)C)CO CC1(NC(c2[nH]ccc2C2CC2)=O)CCCCC1C(=O)NCc1nc[nH]n1 N1(C(CNS(NC)(=O)=O)=O)CC(NC(=O)C=Cc2cccs2)C(C)C1 c1(C(N(CCC)CCNC(C2CCC2C)=O)=O)cc(C)c(Cl)cc1OC N1(C(C(C=C)O)=O)CC2CCC1C1CN(C(C3(n4ccnn4)CC3)=O)CC21 c1(CNC(CCOC)(C)c2nnnn2C2CCCC2)ccc2c(c1)C(=O)NCC2 C1(NC(=O)CC2CCC(C3CC3)O2)CC2(C1)CC2NC(=O)CC1(N(C)C)CCCC1 Cc1cc(C(=O)N(C2CN(C(=O)CC(C)NC(N)=O)C2)C)c(N)cc1F C1(CC(=O)OCC)OCC2CN(C(c3occc3Br)=O)CCC12.C12CCN(C1)C2 c1(C(=O)NC2CCCC2CNC(C2CCCC3(CC3)C2)=O)cc2ncccn2n1 c1(C(C(=O)NC2CC(CNC(=O)CC3(CSC)CC3)C2)N(C)C)ccc(Cl)cc1 C(=O)(C(CC)CC(C)C)NC1CC(NC(C(CC)=CC)=O)C(O)C1 N1(C(CC(=O)OC(C)(C)C)=O)CCC2(CCN(C(C3(C)CC(=O)N(C)C3)=O)C2)C1 c1(C2(C)CC2)cc(C(=O)NC(CNC(=O)Cn2cc(CO)nn2)CO)no1 N1(C(CSCC=C)=O)CCC(CNC(=O)CC(C=C)c2ccc(OC)cc2)CC1 CCCCC(C(=O)N1CCCC1CCNC(=O)C(C)NC(N)=O)NC(N)=O Cc1ccc(CO)c(OCCNC(c2cc(C(C)C)n(C)n2)=O)c1 c1(C(N2CC(CNC(C(CC=C)C)=O)CC2(C)C)=O)ccc2c(C)noc2c1 CCCC(C)(CC)C(=O)NC1CCN(CCCNC(=O)C(F)(F)F)CC1O C1(C(=O)NCCN2CCC(NC(c3scnc3C)=O)CC2)(OC)CC2CCC1C2 C=C(C)CCC(C)NC(c1cnc(CNC(=O)C(C)(C)Cl)nc1)=O c1(C(N2CC(C)(C)C(NC(=O)C=C3CCC3)C2)=O)ccc2cccnn12 Cc1cccc(C2(C(=O)NCC3CC3NC(=O)Cc3cc(C)on3)CCCC2)c1 C(=O)(C1=CC2(CN(C(=O)CC3C(=O)NN=C3C)C2)OC1)N(CC(F)F)CCOC C1(CNC(C(c2ccc(OC)c(F)c2)C)=O)CN(C(=O)C(N)=O)C2(CCC2)C1 c1(C(N(C(CNC(C2CCCO2)=O)C2CC2)C)=O)cccc(S(C)=O)c1 C1(NC(CCc2ncc(C)[nH]2)=O)CN(C(=O)C(C)SC(F)(F)F)C2CCCC12 C1(C(N2CCC2Cn2cc(C3C4CCCCCC34)nn2)=O)CC(O)C12CCC2 S(=O)(=O)(c1ccc(Cl)s1)C(=O)NC(C)CNC(=O)CCCNC(C1CCC1)=O c1(C(=O)NC(CN(C(CC2C(CC)C2)=O)C)C)ncc([N+](=O)[O-])n1C C(N=c1[nH]c2c(c(=NC3CC4(CCCC4)C3)[nH]1)CCCCC2)c1nc(C)c(C)s1 N#Cc1cc([N+](=O)[O-])ccc1NC(C1CC(O)CCN1C(=O)Cc1cscn1)=O C(c1ccc(F)c(Cl)c1)=CC(=O)NCC(CN(C)C(c1cn2c(n1)SCC2)=O)O C(c1cc(F)cc(F)c1)=CC(=O)NC1CC2(CN(C(C3CC(=O)NC3)=O)C2)C1 C#CCCCCCC(C(=O)NCCC)N1CCN(c2ncccc2Cl)CC1 C(=O)(C1CCCc2sccc21)N1CC2CC(CNC(C(C)(C)C)=O)C2C1 C(=O)(C(F)CCC(C)(C)C)NC(C(=O)NC1C(CC)C1)CC1CCC1 CCC(C(=O)N1CCCC1CCNC(c1csc(SC)n1)=O)OC C1(CNC(C2CCCCCC2)=O)CCC2CN(C(c3ccncc3F)=O)CC12 c1(C(=O)NC(COC)C(N2CC(n3ccnn3)C(O)C2)=O)ccc(F)c(C)c1 C=CCCCC(C(=O)NCC=Cc1ccccc1)NC(c1cc(C#N)n(C)n1)=O N1(C(C2CN(C)C(=O)C2)=O)CC(C(=O)NC2CC2C(C)(C)C)CC1(C)C c1(C(=O)NCCN(CCOC)C(C23CCOCC2C3)=O)nccnc1C n1(CC)ncc2c(NC(CNC(C3CC34CCOC(C)C4)=O)C(C)C)ncnc12 C1(C(C)NC(=O)CC2(C)CC2)CN(C(c2ccc(C(F)(F)F)cc2)=O)CCO1 N1(C(=O)NCC(CC2CCCO2)OC)CCN2C(CNS2(=O)=O)C1 C(=O)(C(C)C(C)O)NCCN(CCOC)C(c1sc(Cl)cc1Br)=O c1(CC(=O)N(CCCN(C(C2(SCC)CC2)=O)C)C)c(CC)n[nH]c1CC C(=O)(CC(=O)NC(Cc1cn[nH]c1)C(=O)NCCCNC(N)=O)N(C)C C1(NC(c2c(CC)non2)=O)CC2CN(C(c3cccc(OC)c3F)=O)CC2C1 C1(C(N(CCCNC(C(C)NC(C)=O)=O)C)=O)CCON1C(=O)OC(C)(C)C c1(C(=O)NCC2C(NC(c3[nH]cc(C(C)=O)c3)=O)CCC2)c(F)cccc1F C1(C(=O)NCC(C2CC2)NC(c2cc(-c3cn(C)nc3)on2)=O)CCCCCC1 c1(C(=O)NC(C2CCCCN2C(=O)C2=CCCS2)C)cc(C#N)ccc1Cl N1(C(c2ccc(CC)s2)=O)CC2CC3CC2C1C3NC(c1cc(F)c[nH]1)=O N1(Cc2ccn(CC)n2)CCCC(NC(c2cc(C)on2)=O)C1 C1(C(=O)Nc2cn(CCOC)nc2)CN(C(C2(C)COC(COC)C2)=O)CCO1 CC(CO)CCCNC(=O)CC1CCCN(C(C2C(C#N)C2(C)C)=O)C1 c1(CNC(CNC(C2C(C)C2)=O)=O)ncccc1Cl c1(CC)oc(C(N2CCC(C3CCCN3C(C3C4CCN3CC4)=O)C2)=O)cc1C C(=O)(CC(=O)NC(Cn1cccn1)C(=O)NCCCc1n[nH]c(C)n1)NCC C1(c2cn(C)nc2)CC1N=c1[nH]c(=NCC2CCCCS2(=O)=O)[nH]c2ccsc12 C=CC(C)(CC)C(=O)N1CCC1Cn1cc(C2(C)CCCN2C)nn1 N1(C(c2cnc(CNC(C(CC(C)C)O)=O)nc2)=O)CCC2(CC1)CSC2 c1(C(=O)NC2C(NC(c3cc(CC)nn3C)=O)CCOC2)cccc2nsnc12 c1(OC)cc(N)ccc1C(N1CCC(C)(NC(C2CC(N(C)C)C2)=O)C1)=O Cc1nc(N)c(CC(=O)NC(C)(C)CN(C)C(C2(F)CCOC2C)=O)c(O)n1 N1(C(C2(NC(CN(CCC)C)=O)CC2C)=O)CC(C(=O)OC)OC(C)C1 CCC(CC)C(C)C(=O)NCC1CN(C(c2ccc(C(C)(C)C)cc2)=O)CC1O C=CC(CCC)CC(=O)NCC(O)CCNC(c1cc(CO)n(C)n1)=O C#CCC(C)(C(=O)NCC(C)(C)SC)NC(C1CC2(CCC2O)C1)=O C(C(C)(C)C(C)(C)O)NC(C(CNC(c1c(C)nsc1)=O)N(C)C)=O C(N=c1[nH]c(=NCCc2ncccc2F)[nH]c2c1CSC2)c1n(CC)c(C)nc1 c1(N(C)Cc2c(C)cc(Br)cc2)ncc(S(=O)(=O)NC2(C)CC2)cc1Cl C(=O)(C1=NOC(C)(C)C1)NC(C1CCCCC1)CNC(c1ccc(OC)cc1)=O c1(C(=O)NCC(C)CNC(=O)CNC(N)=O)cccc2[nH]ccc12 Cc1oc(CNC(C2(CN(C)C)CCC2)=O)nc1C(=O)NC(c1nc[nH]n1)(C)C C1(CNC(CSCCCC)=O)COC(CNC(=O)Cc2n[nH]c(C)n2)C1 c1(C(N2CC(SC)C(NC(c3cn(C)cn3)=O)C2)=O)cccc2c1CCS2(=O)=O N1(C(C(C(C)C)c2cccnc2)=O)CCC2CN(C(=O)CCS(C)(=O)=O)CCC12 c1(CN2CCC(C(C)C(N3CCC(C)(C)CC3)=O)CC2)ccc2c(c1)CCC2 C(CCCC(=O)N(C)CCOCCNC(c1cccc(C2CCOC2)c1)=O)=CC CCCC(C)CC(=O)N1CC2CC1CN2c1ncc(C)c(O)n1 N1(C(C23C(CN(C(c4cc(I)c(F)cc4Cl)=O)C2)C3)=O)CCC2(CCCNC2)C1 c1(C(N2CCC(CCOC)(C(=O)OC)C2)=O)cccc(S(=O)(=O)CCO)c1 C1(NC(CC(CNC(c2cc(OC)n[nH]2)=O)O)=O)CCCCC12CC2 C1(CC)(NC(C2CCC(F)C2)=O)CCN(C(=O)CC2=CCCC2)CC1 N1(C(CNC(=O)OC)=O)CCC(C)(NC(C2CN(C)CC2c2cccnc2)=O)C1 CC1CN(C(C2CCC(CN(C)C)O2)=O)CC1NC(=O)CC1CC=CCC1 C=C(C)C1OCCC1C(=O)NCC(=O)NCC(=O)NC1CCCN(C)C1=O n1(CC(=O)NC2(CCC(=O)NC3C(C)(C)CC3)CCC2)cc(C#N)cn1 C(=O)(C(C)(C)S(C)(=O)=O)N(CCNC(C1CC(C(C)(C)C)OCC1)=O)C1CC1 N1(C(c2c(OC)cncc2)=O)CCC2CN(C(=O)C(C)CC(C)C)C2C1 N1(Cc2nc(C)sc2)CC(C(=O)NCCNC(c2ccccc2)=O)CC(F)(F)C1 CC(C(=O)NC1CCC1NC(c1csc(C(F)F)c1)=O)C(C)(C)C c1(C(=O)NC2CCC(CNC(c3ccsn3)=O)CC2)ccnc2ncccc12 N1(C(CCn2c(C)csc2=O)=O)CCCCC2(CCN(CCC3CC3(Cl)Cl)C2)C1 N1(C(Cc2c(C)n[nH]c2C)=O)CC(O)(C2(CNC(=O)C3=CCCCC3C)CC2)C1 c1(C(=O)NC(C2CCN(C(C=Cc3ccc(C)o3)=O)CC2)C)cc(O)cc(O)n1 C=CC(CCC)CC(=O)NCC1(NC(c2nocc2Cl)=O)CCOC1 N1(C(C2N(CC)C(=O)CC2)=O)CCC(C)N(C(c2cc3ncccc3o2)=O)CC1 N1(C(C2C(n3cc(CS(C)(=O)=O)nn3)CCC2)=O)CC2C(Br)C2C1 C1(OC)CCN(C(=O)C(=O)NCC(CSC)OC)CC1 c1(OC)ccc(C(=O)NCC=C2CCN(C(c3sc(C)cc3Cl)=O)CC2)c(F)c1 O=S1(=O)CCN(C(=NCCF)NCC(CO)C2CCOC2)CC1 CC1(C)C(=O)CC1C(=O)NCC1CCCCN1C(C1CCC1)=O c1(C(N(C)CC2COCCN2C(=O)C(O)C2CC2)=O)c(F)cc(F)cc1Cl N1(C(Cc2c(C)scc2)=O)CCC(C)(NC(=O)CSCCC#N)C1 C1(Nc2cc(NCC(C3CCC3)OC)ncn2)CCC(N=[N+]=[N-])CC1 c1(CNC(C2C(OC)CC2)=O)ccnc(N2CCN(C(=O)CCC3CC3)CC2)c1 c1(CC(=O)OC)cccc(C(=O)N(C2CC(NC(c3c[nH]nc3C)=O)C2)C)c1 c1(CC(=O)NC2C=CCN(C(c3cnc(CC4CC4)s3)=O)C2)cccnc1Cl C(=O)(C(F)(F)C(C)O)NC(CCN(C(c1c(C)nn(C2CC2)c1)=O)C)C(C)C C1(CC=C)(C(=O)NC(CN(C)C(C2CCCCN2CCC)=O)CC)CCOCC1 N1(C(C(C)P(C)(C)=O)=O)CCCN(C(c2ccc(N)c(N)n2)=O)CCC1 N1(C(c2cc3sccc3[nH]2)=O)CCC2CN(Cc3cccc(Cl)c3Br)CC12 C1(CNC(C2(COC)CC2(F)F)=O)CC(F)CN1C(c1cc(C(F)(F)F)no1)=O N1(C(COc2cc(C)on2)=O)CCCCC1C1CCCN1C(=O)CC(C)(C)C#N N1(C(c2ccc(OC)nc2C)C(=O)NC2CC(CC)C2)CCC2(CCOC2)CC1 c1(C(=O)NC(C(N2CC(CC)C(F)C2)=O)Cc2ccoc2)cnc(C)[nH]c1=N c1(C(N2CCCC(CNC(c3n[nH]c(C)c3Cl)=O)C2)=O)ccc2[nH]c(=N)sc2c1 N1(C(C(C)(C)CC(F)F)=O)CC2(CCC(NC(C3CC34CCCOC4)=O)CC2)C1 n1(CC)nc(C)c(C(=O)OCC2CCCOC2)c1C(F)(F)Cl c1(C(=O)NCC)cccc(C(N2CCCC(NC(=O)C(COC)OC)C2)=O)c1 C(CC(=O)N(CCF)CC)(C(F)F)NC(C=C(CCC)C)=O N1(C(C(C)C)=O)CCC2(CCCC2CNC(C2CCCCN2C(C)=O)=O)CC1 C1(NC(C(C2CN(C(=O)OC(C)(C)C)C2)O)=O)CCCCC1 c1(C(N(CCCNC(C2CC23CCOCC3)=O)CC)=O)cc2c([nH]1)CCOC2 c1(C(N2CC3C(CNC(C4CCN(C)C4=O)=O)C3C2)=O)ccc(S(N)(=O)=O)o1 c1(C(=O)NC2C(NC(c3cnn(CC)c3C)=O)CCC2)c(F)ccc(O)c1F C1(NC(=O)C=CC(=O)NC2CC2)CN(C(=O)CC2C=CCCC2)C2CCCC12 C(=O)(C(C)S(=O)(=O)C1CCOCC1)NC1CC(CNC(c2occ(C)c2C)=O)C1 C(=O)(CC(F)(F)F)NC1CN(C(C2CCN(C(C)=O)C2)=O)C1 c1(CC)c(C(=O)N(C(C)CCNC(=O)C=Cc2cn(C)nn2)C)nnn1CC C1(C(N(C2CCCN(C(c3c(C)coc3C)=O)CC2)C)=O)C2CCC3C(C2)CC13 CCC(CC)(CC)C(=O)N1CCC(NC(C2CC(=O)N(O)C2)=O)C1 c1(CCC(=O)NCCC(O)COC)ocnc1C(=O)NC(CC)CNC(=O)CO C#CCC(C)(C(=O)N1CCC(C)(O)C1)NC(=O)CCN(C)CCC C=CCC(CC)C(=O)NCCOC1C2CC1N(C(=O)C=C1CCCCC1(C)C)C2 n1(CC)cnc2c(N3Cc4[nH][nH]c(=N)c4C3)nc(=NCCN(C)C3CC3)[nH]c12 C1(O)(CNC(CCCOC(C)C)=O)CCN(C(C2CC2C(C)C)=O)CC1 C(c1ccc([N+](=O)[O-])s1)=C(C(N1CCN(C(C=NOC)=O)C(C)C1)=O)S(=O)(=O)NC c1(C(C)C)ccoc1C(=O)NCC1(F)CC(NC(C2CCOC2C2CC2)=O)C1 C1(NC(CCc2n(C)ccn2)=O)CC=C(C(=O)NCC2CCCC(C)(C)C2)C1 C1(C(=O)NCC(=O)Nc2ccc(F)cc2)COCCN(CC2CCS(=O)(=O)C2)C1 n1(CCC(N2CC(C)C(O)CC2)=O)cnc2ccccc12 C1(CC(N2CCC(C)(CNC(c3nn(CC)nc3C)=O)C2)=O)CCCCC1(F)F C(=O)(C1=COCCO1)N(C1C2CN(C(c3ccc(C(F)(F)F)c(O)n3)=O)CC12)C CN=c1nc(N(C)CCc2ccccn2)[nH]c(=NCCC(=O)OC)[nH]1 C(=O)(C(C)(C)C(C)(F)F)N1CCOCC(CNC(CC(C)(C)N(C)C)=O)C1 c1(CC)nc(C(C)NC(=O)C(=O)NCCC(C)(C)c2ccccc2)n[nH]1 CN1CCOC(C(=O)NCC2CC3CC3N2C(=O)COc2ccc(F)nc2)C1=O Cc1ccc(C(=O)NCCCN2CCC(NC(=O)C#CC(=O)N(C)C)C2)nc1 Cc1cc(C(=O)N(C2CN(C(=O)CCCn3ccnc3C)CC2F)C)oc1C C12(CNC(c3ccc(O)cn3)=O)CCC1CCN2C(C1CCC1)=O C1(F)(CNC(c2c(C)nc(-c3nc[nH]n3)s2)=O)CCCN(C(=O)C(Cl)=CCl)C1 CCCCS(=O)(=O)CC(=O)NCC1C(C)CCCN1C(=O)C(C)O c1(CN2CCN(C)C(CC3CC3c3ccccc3)C2)n[nH]c2ccc(F)cc12 C(=O)(CCCCCSC)NC(CNC(Cn1c(CCC)nnc1S)=O)C Cc1ccc2sc(N3CC(CCCCNC(=O)C(O)CC(C)(C)C)C3)nc2c1 N1(C(c2cnccn2)=O)CC2(CCN(CC3CCCC3N3CCOCC3)CC2)C1 C1(NC(c2cnn(-c3ccccc3)n2)=O)CCCCN(C(c2cnco2)=O)CC1 c1(C(=O)NC2(C3CC3)CCN(C(COC(CC)C)=O)C2)cnc2c(c1)CCCC2 CC1CC(NC(c2cc3n(c2)CCC3)=O)CCN1C(=O)C=Cc1ccncn1 c1(C(=O)NCC2(OC)CN(C(=O)C(F)CC3CCCC3)C2)ccc(N)cc1Cl Cc1cnc(C(=O)NCC2CC2C(=O)NC(CO)C(C)C)c(C)c1 C1(C(N2C(C=C)CC2)=O)CC(C)CN(C(=O)C=Cc2ccc(C)o2)C1 CC1CCCN(C(c2ccc(C3CC3)o2)=O)C1CNC(C1CC(C)(O)C1)=O CC1=C(C(=O)NC2CCCC(CNC(=O)CC3CN(C)C3)C2)CC1 C(=O)(CC(C(F)F)C(C)(C)C)N1CC(CC(C)NC(C2=C(C)OCC2)=O)C1 C1(NC(CC2ON=C(C)C2)=O)CN(C(c2cc(F)cc(Cl)c2N)=O)CC12CCC2 CCCCCCCCC(=O)N(CCNC(C1CCC(O)C1)=O)Cc1ccccc1 c1(C(=O)NC2CC(C(=O)NCC(CSC)(C)O)CC2O)ccc(=O)n(C)n1 c1(SCC(N2C(CC(=O)NC)C(=O)NCC2)=O)ccc(CO)cc1[N+](=O)[O-] N1(C(C)CC(N2CC3(C2)CN(C(=O)Cn2cccc2)C3)=O)CCc2ccccc21 N1(C(c2ccc(CC)[nH]2)=O)CCN(C(c2cccc(CS(C)=O)c2)=O)C(CC)C1 C(=O)(CCS(C)=O)N(C(CNC(=O)C(C)(O)c1ccccc1)C1CC1)C Cc1ccn2c(C3CCN(C(=O)Cc4ccc5nc[nH]c5c4)CC3)nnc2c1 c1(NS(C)(=O)=O)ccc(C(=O)NCC2(CNC(C3CNC(=O)N3)=O)CC2)c(Cl)c1 c1(C(N2C3C(NC(Cc4nc(C)sc4C)=O)C(C3)C2)=O)cc(F)c(F)c(Cl)c1F c1(C(N2CCC(CC)C2CNC(=O)CN2CCSCC2)=O)n[nH]c2c1CCC2 C(=O)(C1=CCCCC1C)NCC(=O)NC(c1nnc(C)o1)C Cc1c(C(N2CCCC(C(C)NC(c3cn4c(n3)SCC4)=O)C2)=O)cccc1N c1(C(=O)NC(C)(C)CCNC(C2(c3cc[nH]n3)CC2)=O)cc(Cl)cc(Cl)c1F N1(C(CC=C)=O)CCC(C2CCN(C(=O)CC(F)(F)Br)CC2)C1 Cc1ccncc1C=CC(=O)NC1CN(C(=O)CO)CCC1c1ccccc1 c1(OC)cc(C)c(NCCCCSC)c(C)c1 c1(C(=O)NCCCCNC(C2C(C)(Br)C2)=O)ccc2c(c1)C(=O)OC2 c1(C(N(CC(C)NC(Cc2ccc(C(C)=O)nc2)=O)C)=O)nccc(Cl)c1F CC1(C#CC(=O)NC2CCN(C(c3cc4n(n3)CCO4)=O)C23CC3)CCCO1 Cc1snnc1C(=O)NC1(CNC(C2(O)CCOC2)=O)CC1 C(CC(C)C)(C(=O)NC1CC2(C1)CN(c1ccnc(-c3ccccc3)n1)C2)OC c1(C(=O)NCC2CCCC(CNC(c3n(C)ncc3Cl)=O)C2)cccc(F)c1N c1(CCC(=O)NC2CN(C(c3ccc(Br)o3)=O)C2)cncc(O)c1 Cc1ccc(C(N2CCCCC2CCN(C(=O)C(C)CC(C)C)C)=O)c(C)c1Br C1(CC(=O)NC(CC=C)(C)C)CC(C)N(C(=O)C=Cc2cc(C)no2)C1 C1(N(CCOC)C=O)CCN(C(N)=O)CC1.C1CN(C(=O)CCOC2CC2)C1 N1(C(C(C)OCCC#C)=O)CC2CC(NC(=O)C(C)(C)C#N)C(C2)C1 c1(CC(N2CC(CCNC(COCC3(CC)CCC3)=O)C2)=O)c(O)ncnc1O c1(C(=O)NC2C(C)CN(C(c3coc(CO)c3)=O)C2)cnc2cc(O)ccc2c1 N1(C(CC2ON=C(C)C2)=O)CCCC12CCN(C(c1cc(O)ccc1C)=O)C2 C1(C(N(CCN(C)C)Cc2nccs2)=O)(C(=O)OC)CC2(CCC2)C1 Cn1ncc(S(C)(=N)=O)c1C(C1CCN2CCOCC12)N N1(C(c2c(CC)ocn2)=O)CCC(C(C)NC(=O)C(=O)NCCC(N)=O)CC1 Cc1cc(C(=O)NCC(O)CNC(=O)CC2CCSCC2)nn1C(C)C c1(OC)csc(C(N2CCC(C(C)NC(c3cscc3C(F)F)=O)C2)=O)c1OC c1(C(=O)NCC2CN(C(c3nnc(C(F)(F)F)s3)=O)CCO2)ccc(F)c(Cl)n1 N1(C(CC(=C)C)=O)CC(N(C(=O)CCc2ccc(CO)cc2)C)C2(CC2)C1 C1(CN)CCc2nncn2C1.C12CCCCN1N(C1CCS(=O)(=O)C1)c1nc2n[nH]1 c1(C(N2CCC(NC(=O)Cc3cc[nH]n3)C(F)C2)=O)ccc2c(c1)S(=O)(=O)NC2 C(=O)(C1CCCc2cncn21)NC(C(C)C)CNC(c1cc(Cl)ccn1)=O c1(CC)cccnc1C(=O)NCC1(C)CCN(C(c2cc(C)nn2C(F)F)=O)C1 n1(CC(=O)N(C(C)C)C2CC2)cc(CNC(c2ccon2)=O)nn1 N1(C(c2c(C)cc(Br)cn2)=O)CC2(CCC2)CC1CNC(c1cocn1)=O c1(C(=O)O)cc(NCCc2ccc(Cl)cc2F)cc(S(=O)(=O)NCCO)c1 C1(C(=O)NCc2n(CC)nnc2C)CCC(C)(C)N(C(C2(CO)CC2)=O)C1 N1(C(CN(C(=O)CCC2CC2)CC=C)=O)CC2CC(NC(=O)CO)C(C2)C1 C1(NC(C)=O)CCCN(C(C2CN(C(C3CN(C)CCO3)=O)CC2C)=O)C1 c1(NC)ccc(C(N2CCC(NC(C3CCC3(F)F)=O)C(O)C2)=O)c(Cl)c1 Cc1cc(C(F)(F)C(=O)NCCN(C(=O)CCCn2ccnc2)C)cnc1Cl c1(C(=O)NC(C)CCCNC(=O)C(=O)N(C)C)cc2ccccc2cn1 C(=O)(C1CCCc2nc[nH]c21)N(C1CCN(C(=O)C=Cc2cn(C)cn2)C1)CC C1(C(N2CC(COC)N(C(=O)CCc3ccoc3)CC2)=O)Cc2cccnc2C1 c1(C(=O)NCC2OCCCN(C(C=C(C)C)=O)C2)cnn2ccccc12 c1(C(N(C2CC(NC(=O)C(F)CC3CC3)C2)C)=O)cc(Br)ccc1Cl C=CC(C)(O)CC(=O)NC1CCN(C(=O)CCC(=O)NCC)CC1 N1(C(C)=O)CCCCC1c1nc(Cc2ccccc2F)nn1CCOC(C)(C)C c1(C(=O)NC(CC)CNC(=O)CC(C)C)coc2c1CSC2 c1(C(N(CC(C)NC(=O)CCc2cnn(C)n2)CC)=O)ccc(F)cn1 C1(NC(C2CCCC(F)C2)=O)C=CCN(C(c2ccc[n+]([O-])c2)=O)C1 N1(C(C2(C(=O)OC)CC2)=O)CCCC(C2CCCCN2C(=O)Cc2nocc2C)C1 c1(CC)ccc(OC)cc1C(=O)NC1CCC12CN(C(c1cccc[n+]1[O-])=O)C2 c1(C(N(C)CCN(C)C(C2CC(O)CN2C)=O)=O)ccccc1[N+](=O)[O-] N1(C(C(C)(C)OCC)=O)CCCC(Cn2cc(C(C)(C)OCC(=O)NC)nn2)C1 CC(CCNC(C1CC(O)CCN1C(c1nn(C)cc1Cl)=O)=O)CC(C)(C)C c1(C(CNC(C)=O)NC(=O)C(Cl)=CCl)ccc(C)cc1 C(CC(C)CCNC(=O)CN1CCC(C)(C)C1)NC(C(C)C1CCC1)=O N1(C(c2cn(CCC)nn2)=O)CCCCC2C1CCCN2C(c1ccncc1)=O C1(NC(C2CCC(CCC)CC2)=O)CCN(C(=O)C(C)COC(C)=O)CC(O)C1 c1(NC2CC3(CN(C(=O)OC(C)(C)C)C3)C2)cccc2oc(O)nc12 C1(OC)CC2(C1)CC(C(N1CCC(CNC(=O)C(O)CN3CCCC3)CC1)=O)C2 c1(C(N(CC(O)CNC(c2cc3c(s2)CCC3)=O)C)=O)nc(O)nc(O)c1F CC1CN(C(c2nccnc2Cl)=O)CCC1CNC(c1ncc(Cl)cc1Cl)=O c1(C(=O)NCC(C)N(C(C2N(C(=O)NC)CCC2)=O)C)cnc(O)cc1OC Cc1cc(F)c(NC(c2ccc(SCC3CCCC3)cc2)=O)cc1Cl c1(CC)ccc(Br)cc1C(N1CCC(NC(=O)C2=NOCC2)C(O)C1)=O c1(C(N(C2CCN(C(CCC(CC)CC)=O)C2)C)=O)cc2ccc(OC)cc2s1 Cc1nc(NCC(C(C)C)N(C)C)cc(=NCc2noc3ccccc23)[nH]1 Cc1cc(C)n(C(C)C(=O)NCC2CCCN2C(c2cnn(C(F)(F)F)c2)=O)n1 c1(OC)cccc(C(N2CC(CCNC(=O)C(C3CCOC3)OC)C2)=O)c1F c12cccc(c1O)NC(=O)C1CCC(C1)NC2=O.c1(CC)ccc(NC=O)cc1 N1(C(C(C)C)=O)CC(CNC(C2CC2F)=O)C2(CCOCC2)C1 C=C1CC(C(N2CC(CC(C)C)C2)=O)(CNC(c2sncc2C)=O)C1 C1(NC(c2n(CC=C)nnn2)(C)CSC)CC2(C1)CC(C)C2 C1(CNC(C2(COC)CCOC2)=O)CN(C(c2cn(C3CC3)nc2C)=O)CC1O C(=O)(C(C)S(C)(=O)=O)NCCN(CCC)C(c1ccc(CO)cn1)=O c1(C(=O)NCCN(c2nc(C3CCCCC3)cs2)CC2CC2)ccc2sncc2c1 C=CCC(CC(F)F)C(=O)N1CC2CN(C(=O)C3=CCCC(C)(C)C3)CC2(C)C1 C1(OCC)CC(NC(=O)C(C2(O)CCCCCC2)F)C12CCOCC2 c1(C(N(CCCNC(CC2(OC)CCC2)=O)C2CC2)=O)ccc(C)o1 S(=O)(=O)(c1cccc(C(=O)OCC23CC(C)(CO2)C3)c1)NC(CC)C C#Cc1ccc(F)cc1C(=O)NC1CN(C(c2cc(CC)ccc2F)=O)C1 C1(NC(c2cc(O)nc(O)n2)=O)C2CCC(C2)C1C(=O)NC1CCCCC12CC2 C1(C(N2CCC(C)(CC(=O)Nc3ccc(OC)nc3)C2)=O)CCCC12CCC2 C=CCCN=C(NCc1ccc(C)cc1OCCCC)NCC(C)(O)C(F)(F)F N1(C(C(C=C)(C)CC)=O)CC2(CCN(CC(=O)NC(C)C)C2)C1 c1(C(=O)NC2CN(C(C3OCCN(C)C3=O)=O)C2)nc(C2CC2)n2ccccc12 C1(Nc2cnn(CC)c2C)CCC(F)(F)CC1.n1(C(CC)C)nnnc1CC1CC1 CC1CCN(C(=O)C(=O)Nc2ccccc2)C1c1cn(C2C=CCCC2)nn1 N1(C(C(CSC)C)=O)CCC2(C1)CN(C(=O)C(C)Sc1ccc(F)c(F)c1)C2 C=C(C)CC(C(=O)NC1C=CC(CNC(c2cc(C3CC3)no2)=O)C1)OC C=CCCC(C)(C)C(=O)NC1CC2CCC1N(C(=O)C(F)(F)C(O)CC)C2 c1(OCCC(=O)NC2C(C)CN(C3CC3)C2)ccc2c(c1)OCO2 c1(OC(C)(C)C)ccccc1CC(=O)NCC1CC(NC(C2(C)CC2F)=O)C1 N1(C(c2c(C)nsc2)C(=O)NC2CCCC2)CCN(C)CC1C(C)C c1(CC)ncccc1C(=O)NC1CCN(C(c2cc[nH]c2CC)=O)C1C1CC1 c1(CC(=O)NC2CC(N(C)C(c3ccc(OCCO)cc3)=O)C2)cc(F)cc(F)c1 C1(CNC(C(C)Cc2ccnn2C)=O)(CNC(C2(C)CCCC2)=O)CC12CCC2 Cc1cn2nnc(C(=O)NCCCN(C(C3C4CC(=O)CC34)=O)C3CC3)c2c(O)n1 c1(C(c2n(CCCSCC)nnn2)NCC2CCCOC2)cc(S(C)(=O)=O)co1 C(=O)(CC(CC(C)C)NC(c1ccnn1CC)=O)N1CCOCC(=C)C1 C1(NC(C(C)CC)=O)CC2CCC1N(C(c1cc(CC)nnc1C)=O)C2.CCC C(=O)(C(C(C)C)n1cnc(C)c1)NCCC1N(C(c2c(CC)nc[nH]2)=O)CCC1 C(=O)(C(CNC(c1ccsc1Cl)=O)N(C)C)N(C1CCN(C)C1)CCC C12(NC(=O)CCN3CCCCC3=O)CCC1CN(C(C1CCCCC1)=O)C2 C(=O)(C(F)CC(CC)CC)NC(CCCC)CNC(=O)CCc1ccccc1F C(=O)(C(C)(C)N=[N+]=[N-])NCCC1C(C)CN(C(c2cc(O)ncn2)=O)C1 C1(C(=O)NCC2CCC(NC(c3cn(C)nc3O)=O)CC2)CN=C2N=CNN2C1 c1(C(=O)NC(C)CNC(=O)CCc2ccccc2)cc2c(nc1O)CCSC2 CC1CC(C)CN(CCCNC(=O)OC(C)(C)C)C1.C1(=O)C(O)CCN1 c1(-c2cn(C(C(=O)NCC(C)C)C)nn2)ccccc1OCC(=O)O C1(CNC(c2c(CC)cco2)=O)CC(NC(C2(O)CCOCC2)=O)CC1O N1(C(CCCC(=C)C)=O)CC2CC(C)N(C(c3ccc(N(C)C)cc3)=O)C2C1 N1(C(c2ccc(CC)o2)=O)CC(CNC(C2CC(CC3CC3)C2)=O)CC12CCC2 C1(C(N2CCC(C(C)C(=O)NCC=C(Cl)Cl)CC2)=O)CN(C)CCN1C CC1CCc2nc(Cl)nc(N3CC(CN(C)C(C4(C)CC4)=O)C3)c2C1 c1(CC(C)C)c[nH]c(C(=O)NCC(C)CNC(=O)CN2CCC2C)c1 c1(OC)ccc(C(=O)NCC(C)NC(=O)Cc2cc(C)ccc2F)n2nccc12 c1(C(N(C(C)CCNC(c2cc(C(F)(F)F)cs2)=O)C)=O)cccnc1F n1(CC(C)C)ccc(C(=O)N(C2CCCC2)CCNC(=O)C=Cc2ccsc2)n1 CC1(C#CC(=O)N2CCC(CF)(NC(=O)CC3C=CCC3)C2)CCCO1 c1(C(=O)NC2CCN(C(c3cnc(CCC)s3)=O)C2)ccc2c(c1)CCN(C)C2 C1(c2nnnn2CCCC2CC2)(NCc2ccn(C(C)(C)C)c2)CCC2CC12 N1(c2nnn(C)n2)C2CCCC1CN(C(=O)Cc1c[nH]c3cc(Cl)ccc13)C2 Cc1cccnc1CN(C)CC1CCN(C(=O)CNC(=O)Nc2cccs2)C1 CC(=O)CCCC(=O)NC1CC2CC1CC2C(N1CCC(C2CC2)C1)=O C(=O)(CCCN(C)N=O)N(CCOCCNC(C(CC=C)C)=O)C C(=O)(C1=C(CC)OCCS1)N1C(CCCC)CN(C(=O)C(F)C2CC2)CC1 C1(C(N(C(CC)C2CC2)C)=O)CCN(C(=O)NC2CCCO2)CC1 C(c1cncnc1O)=CC(=O)NC1C(OC)CN(C(=O)CC2(O)CCCOC2)C1 Cn1nccc1CCNC(c1cc(CNC(=O)C=CCN2CCCC2)no1)=O N1(C(CC(COC)COC)=O)CC2(C1)OC1(C)CC2(NC(C2CCCOC2)=O)C1 CC(CS(C)=O)C(=O)NC(C)(C)CCC1CCN(C(C2CCS(=O)CC2)=O)CC1 c1(C(N2CCC(CNC(C3(C#N)CC4CC4C3)=O)CC2)=O)nnn2c1COCC2 N1(C(c2ccc(C)nc2O)=O)CCC2CCCN(C(c3cc(Cl)n(C)n3)=O)C2C1 N1(C(c2cc(C)cc(O)c2)=O)CCCC1C1CCCN1C(=O)CN(C)S(N)(=O)=O c1(C(=O)NC(C2CN(C(CN(CCOC)C)=O)C2)C)ccc(C2CC2)nc1 N1(c2c(C#N)cncn2)CCOC2CN(C(c3cnc(O)c(Cl)c3)=O)CC12 C(c1ccc(NC(C)=O)cc1)=NC(c1ccc(CNC(CSCC#C)=O)cc1)=O c1(C(N2CCCC2c2cn(Cc3cnoc3)nn2)=O)ccc(-n2cnnn2)cc1 c1(C(=O)NC(C(C)NC(c2c(OCC)cccn2)=O)CO)nsc2ccccc12 C(=O)(CCCC(C)=O)N1CC2C(CNC(c3c(CC)nc[nH]3)=O)(C2)C1 c1(NCCOCCNC(CC2CCC(C)O2)=O)ncnc2c1ncn2C1CC1 N1(CC)C(=O)NC(c2ccc(N)c(Br)n2)C2=C1C(C)CN(C)C2=O N1(C(Cc2c(C)noc2)=O)CCC2CCN(C(c3ccc4c(c3)CCN4)=O)CC12 C=CCC(CC(C)C)C(=O)N1CCN(C(c2cccc(N)c2O)=O)C(COC)C1 CCC(C(=O)NCC(C)NC(C1SCCS1)=O)SC C1(NC(c2cccc(-c3ccncc3)c2)=O)COCCN(C(=O)CC2CC2)C1 c1(C(=O)NCC(C)N(C)C(c2csc(-c3nc[nH]n3)n2)=O)cc2n(c1)CCCC2 CC(C)C(CC(=O)N1CCCCCC1)NC(=O)C(CO)N(C)C O=C1NC(=O)CN1.N1(C(CCn2cc(C)nn2)=O)CCC(C(O)C(F)(F)F)CC1 CC1C2C(CCN2C(=O)CNc2cccnc2)CN1C(=O)C1=COCCO1 C1(C(N2CC(C)(NC(c3c(C(=O)OC)scc3)=O)C2)=O)CC2CCCCC2O1 C1(CC(N2C(CO)CC2C)=O)(OC)CN(C(=O)Cc2cc(C)on2)C1 N1(C(=O)OC(C)(C)C)CCC(O)C(NCc2ccc(Cl)nc2Cl)C1 N1(C(C2CSC2)=O)CCC2(CC1)CC(n1cc(CO)nn1)CCO2 C(=O)(C(CC(C)C)N(C)C(C1CC(=O)CCO1)=O)NCCc1scc(C)n1 c1(OC)ccc(F)c(CN2C(C(=O)N(C)CCC3OCCO3)CC3CC23)c1F N1(C(c2cccc(CC)c2)=O)CC2CCCC2(NC(=O)CCc2cncnc2)C1 CN1CC=C(CC(=O)N2CCC3CCC(C2)N3c2nc(C3CC3)nc(Cl)c2C)CC1 N1(C(Cc2scc(C)c2)=O)CCCC(O)(CN(C(=O)Cc2ccns2)C)C1 S(=O)(=O)(c1ccc(C#N)c(NCc2c[nH]ccc2=N)c1)NCC1C(C)OCC1 CC1CN(C(=O)CSc2ccc(F)cc2F)CCC1CNC(c1cnsc1)=O CON(CCC(=O)NC(C(=O)NC)C1CCOC1)C(=O)C(C)N1CCCC1=O C1(C(N2CC(OC)C(NC(=O)CC(Cl)Cl)CC2)=O)CC12CCC(=O)CC2 c1(OCC)ccc(C(N2CCCC(CNC(=O)C(C)COC)C2)=O)cc1C c1(CNC(C2C(CC)NCC2)=O)cc(C)ccc1C C1(O)(CCC)CCN(C(C2CN(C)CCN2C(C2CCSC2)=O)=O)CC1 c1(C(=O)NCC2(O)CCN(C(CCC(=O)OCC)=O)C2)ccc(C)c(C)c1Cl c1(C(=O)NC(CNC(c2[nH]cc(C(C)(C)C)c2)=O)C2CC2)ncn2c1CCC2 C(=O)(C(C)CC(C)C)NCC1CN(C(c2c(CC)n(C)nc2)=O)CC1C c1(C(=O)NC(C2CC2(C)C)CC)ccc(CNC(c2cnc(CC)s2)=O)cn1 CC(CCN=c1[nH]c(N2CC3CCN(C)CC3C2)nc2cc[nH]c12)c1cn[nH]c1 C1(CC)C(C(=O)NC2CC3(CCCC3)C2)CCCN1C(=O)CCC(C)N(C)C N1(C(C(C)(CO)NC(C(=O)N(C)C)=O)=O)CCOC2CCC12 C(=O)(N=c1[nH][nH]c2ccc(C(=O)O)cc12)N1C(C(C)C)C2(C1)CCOCC2 C1(n2cc(C(C)NCCC=C)nn2)CCC(OC)CC1.C1C(SC)C(=O)N1.OC c1(NC(C2C3CN(C(c4c(CC)occ4C)=O)CC32)=O)cc(O)ccc1C N1(C(CCOC)=O)CC(NC(c2ccc(Br)c(F)c2N)=O)CC12CCOC2 C1(C(=O)NC2CCC(NC(c3cnn[nH]3)=O)C2)(CN(C)C)CCCC1 Cc1cc(C#N)ccc1C(=O)N(C1(C(=O)NC2C(=O)OCC2CO)CC1)C N1(C(C(N2CCSCC2)C)=O)CC=CC(NC(=O)C(c2ccnn2C)O)C1 N1(C(C(COC)N(C)C)=O)CCCC(CC(=O)Nc2cnn(C)c2C)C1 N1(C(C(C)n2ccnn2)=O)CC2CCCC(C1)N2C(=O)CC1CCN(C)CC1 N1(C(c2c(C)scn2)=O)CCC(O)(C(C)NC(=O)CC(C)C(F)F)CC1 c1(C(=O)NC(CNC(CC(C=C)(C)C)=O)(C)C2CCC2)ccc(N)c([N+](=O)[O-])c1 C1(C)(CNC(C2(SCC)CC2)=O)CN(C(=O)CC2CCCOC2)CCO1 C12(NC(C(N3CCCCC3=O)C)=O)CC1CN(C(=O)CCc1cc[nH]n1)C2 C12(NC(c3cc(Cl)ccc3F)=O)CCN(C(c3conc3C3CC3)=O)CC1C2 N1(c2ncnc(NC(CCC)c3ccco3)c2C)CCCN(C)C(=O)C1 c1(C(CNC(C=CC(C)C)=O)NC(c2cccn2C)=O)ccc(F)cc1 N1(C(c2cc(C)oc2C)=O)CCC(NC(=O)Cc2cc(F)ccc2O)CC1C c1(C(C(=O)NC(C)(CNC(=O)C=C2CCC2)C2CCC2)=O)ccc(F)cc1 Cc1[nH]c2ccc(C(=O)OCc3ccc(C(F)F)c(F)c3)cc2c1C C(CC1=CCN(C(=O)CC2CCCCC23CC3)CC1)NC(C1(C)CCOCC1)=O CC(C)(C)C#CC(=O)N1CCN(C(=O)CC2CCCOC2)CC1c1ccccn1 C1(O)(C(N(CCCNC(c2ccc(CCF)cc2)=O)C)=O)CC2CCC1C2 C=CCC(CNC(c1nnn(C)c1C)=O)C(=O)NCC12CC(CN1C)C2 c1(OC)ccc(Cl)c(CC(N2CC3C(NC(C4CC4F)=O)C3C2)=O)c1F c1(COC)nc(C)c(C(=O)NC2C=CC(CNC(c3cscc3C(F)F)=O)C2)s1 C(=O)(CC(C)(C)C)N(C(C)CNC(c1cnn(C2CCC2)c1)=O)C C(=O)(C(O)CC(N)=O)N1CCC(NC(=O)NC2(CC)CCOCC2)C1CC N1(C(C(C(C)C)C(=O)NC(c2ccc(OC)nc2)=O)=O)CC2(CCCCCC2)C1 c1(CC(=O)NC2C(CNC(CN(C3CC3)CC)=O)CC2)c(Cl)cccc1Cl C=CCCCC(C(=O)Nc1cnc(OC)nc1)N(C)CCC1CC1 c1(C(=O)OC)ccnc(CSCCS(C)(=O)=O)c1 N1(C(c2c(C)nncc2)=O)CC2(C1)CN(C(C1(C)CCCS1)=O)C2 CCC(CC)C(F)C(=O)N1CCN(C(c2ccc[nH]2)=O)C(c2ncc[nH]2)C1 c1(C(C)C)n[nH]c(=NCCC(C)NC(=O)C(C)(C)CO)o1 C(C(C(=O)NCC(O)C(=O)NCCC1CCCC1O)N(C)C)N(C)C c1(OC)ccc([N+](=O)[O-])cc1CNC(c1ccc(I)cc1)(C)C c1(CC)n[nH]c(=Nc2cccc(F)c2C(=O)NCC(C)(C)O)o1 c1(CC=C)cccc(CN2CCCC(C(N3CCC4(CC4)C3)=O)C2)c1O c1(CC)ncc(C(=O)NCC2CC(F)(CNC(=O)CCCC#N)C2)c(C)n1 c1(COC)nc(C)c(C(=O)OC)c(O)n1.C12CC1N(OC(=O)CC(C)C)C2 N1(C(C2(c3cc(C)no3)CC2)=O)CC(NC(=O)CNc2ccccc2)C(C)(C)C1 Cc1cc(C(F)(F)F)c2cc(C(=O)NCC(C)(O)C(C)C)oc2n1 C1(NC(C(CC)N(CC)CC)=O)COC2(C1)CN(C(=O)CC1OCCO1)C2 c1(N2CCC(C)(CCO)CC2)ccc(S(=O)(=O)N2CCCC(F)C2)cc1Br Cc1cn(C)nc1CNC(=O)N(C1CC(c2ccccc2)C1)C c1(C(=O)Cc2cccc(C(=O)OC)c2)ccc2c(c1)CCCC2.C12CN(C1)S2 c1(C(=O)NC2CC3(CCN(C(=O)CCC4CCC4)C3)C2)cc2cc(Cl)cnc2o1 Cc1c(NC(C2CCCCC2C)=O)nnn1Cc1ccncc1 N1(C(C2CCC(C)O2)=O)CC2(C1)CN(C(=O)Cc1cn(CCO)nn1)CCO2 C(=O)(CCC(C)C#N)N1CC2C(CNC(CCc3cncc(OC)n3)=O)(C2)C1 c1(C(=O)NC(C2CCN(C(C(C)OCC#C)=O)C2)(C)C)ccc(OC)c(F)c1F CS(=O)CCC(=O)NC(C)(C)CNC(c1cc(C2CCOCC2)[nH]n1)=O C1(NC(C2CC3(CCC3)CO2)=O)CC2(CCCN(C(C3CCCCC3O)=O)C2)C1 c1(C(=O)NCC=CCNC(CC2C(C)(C)C(O)C2)=O)cc2ccc(O)cc2[nH]1 C1(Nc2cc(C)nc(N3CCC(c4coc(=N)[nH]4)CC3)n2)CCCCC(F)(F)C1 c1(C(=O)NCCC2CN(C(C(CCC)NC(C)=O)=O)C2)[nH]nc([N+](=O)[O-])c1Cl Cc1cc(F)c(C(=O)NC2CC3CC2N(C(=O)CCN2CCCCC2)C3)c(F)c1 c1(OC)cncnc1NC(C1CCN(C(c2snc(Cl)c2Cl)=O)CC1)(C)C C1(CCNC(CSCCOC)=O)CCCC(NC(=O)COCC(C)(C)C)C1 C1(NC(c2ccc(-c3ccccn3)o2)=O)CCC12CN(C(=O)CC1OCCO1)C2 c1(C(=O)NCC2(OCC)CN(C(=O)C=Cc3ccccn3)C2)cc(C#N)c[nH]1 C1(C(N(CCCNC(CS(CC)=O)=O)C)=O)CCc2nc(C3CC3)ncc2C1 C(=O)(CC(C)C(C)(C)C)N1CC(NC(CCCOCCC)=O)C(n2ccnn2)C1 C(N=c1[nH]nc(CC(C)C)s1)C1CCC(NC(c2c(NC(C)=O)cccc2)=O)C1 c1(C(=O)NC2CC3CN(C(C(=O)NC(C)C)=O)CC32)cccc2ncnn12 C1(NC(c2c(C)nccc2)=O)CC2CCC1N2C(C1(C(C)(C)C)CCCCC1)=O c1(OC)cc(C(=O)NC2CN(C(=O)Cc3cccc(F)c3)CC2C#N)cnc1Cl C1(C(=O)OCC)CN(C(C2CNC3(CCC3)CO2)=O)c2cccc(Br)c2O1 N1(C(C2C(C)(C)C2)=O)CCC2(C1)CN(C(C13CCC(C1)C(C)(C)O3)=O)C2 C(=O)(C(F)CCC(C)(C)C)NCC(C(=O)NC(C)C1CC1)CC1CC1 C1(CCNC(C(C2N(C(Cn3ccc(C)c3)=O)CCC2)(C)C)=O)CCCCCC1 C(CS(=O)(=O)N(C)Cc1cc(OC)ns1)(c1ccccc1)OC C(N=c1[nH]c(=NCc2nnn(C)n2)[nH]c2cccnc12)C1CCn2c(C)nnc2C1 C12(CCC(=O)NCC3(CN(C(C(CC)O)=O)CC)CC3)CCC(CC1)C2 N(C1c2ccccc2CC1NC(=O)CC1CCC1)C(C(C)c1cc[nH]n1)=O c1(OC)ccc(Br)c(C(N2CCOC(CNC(=O)CC(O)C(C)C)C2)=O)c1 O=C(C(CO)C(F)(F)F)NC1(C(=O)NCC2CC23CCOCC3)CC1 N1(C(c2c[nH]c(=N)o2)=O)CCN(C(C2CCCS2)=O)C(c2ccc(F)cc2)C1 C(=O)(C(C)(C)CNC(=O)Cn1cc(Cl)cn1)NC1C(OC)COC1 C(=O)(C(C)CC(C)CC)NC1CCN(C(COc2cccc(C#C)c2)=O)C(C)C1 CC1CC(C)(C(=O)NC2(CNC(=O)CNc3ccccc3CO)CC2)CC(C)O1 C1(CNC(C(C(C)C)NC(=O)OC(C)C)=O)CCN(C(c2ccoc2)=O)CC1C n1(C(C)C)nnc2c(NCCC3CCN(C(=O)C(C)CN(C)C)C3)ncnc12 C1(CC)CN(C(C2CC23CCOCC3)=O)CCC1NC(c1ccncc1F)=O n1(CC(=O)N(CC#C)C(C)C)cc(CNC(C2CCCC2C)=O)nn1 C1(CNC(C=CCN(CC)CC)=O)(NC(C2(F)CCCC2)=O)CCCC1 CC1CCC(O)C(NC(=O)CC2CC(NC(=O)CC3CC(C4CC4)C3)C2(C)C)C1 C1(C(=O)NC2CC(CNC(C3C(CC)N(C)CC3)=O)C2)CC2CCC(C1)C2 N1(C(CC(CC)SC)=O)CC2CCC(C1)N2CCC(=O)NC(C(=O)NC)C(C)C C1(C2CC2)(C(=O)NCCC2CCN(C(CNC(C(CC)C)=O)=O)C2)CCOCC1 c1(C(N2CCC(OC)(CNC(C)=O)C2)=O)cc2c(Br)ccc(F)c2[nH]1 c1(OC)cccc(CC(=O)NC(C2(O)CN(C(=O)CS(=O)(=O)N(C)C)C2)C)c1Cl CC(C)C(F)(CNC(c1cncnc1O)=O)C(=O)NCc1ccc(C#N)s1 c1(CC)cc(C)nc(NC2(CO)CCN(C(C3CCC(N(C)C)CC3)=O)CC2)n1 C(CC1CC1)(C(=O)NC(Cn1cncn1)C(=O)NC1CC(OC(C)C)C1)OC c1(C(=O)NCCC(C)N(C(c2c(CC)ccs2)=O)C)ccc(C(C)C)c(C)c1 c1(C(N(CCN(C(CCC(=O)NC)=O)C)C)=O)nc(C(C)C)ncc1Cl CCS(=O)c1ccccc1C(=O)NCCNC(=O)CNC(=O)C(C)n1cccn1 C(C(C(=O)N1CCC1(C)CCO)n1cc(C(C2CCOCC2)C)nn1)OCC C1(CN(C)NC(C2CC3(CCCC3)C2)=O)CCOCC12CCC2 C(=O)(C1=C(C(F)Cl)N(CC2CC2)C(=O)NC1c1cc(I)c(Cl)cc1F)OCC C(C1CCOCC1)=CC(=O)NCC(CCC)NC(c1cc(C)nn1CC)=O N1(C(CC(CC)C)=O)CCC(C)(C)C(NC(c2cc(C(C)C)[nH]n2)=O)C1 N1(C(c2c(CC)ccs2)C(=O)NCCSC)CCCCCCC1 c1(N(C)C)ccc(-c2noc(-c3cn(C4CCCC4)nn3)n2)cc1N(C)C C1(C(=O)NC(CCC)CNC(=O)COC2CC=CC2)CCCCC1CC CCCC(CCCNC(=O)C(C1CC1)OC)NC(=O)C=CC(F)(F)F c1(CC)ccc(C(=O)NCCC2CN(C(=O)C(c3cncn3C)O)C2)s1 Cc1cc(C(N2CC(NC(=O)C(C)(O)CC(F)F)C(C)C2)=O)c(O)nc1C C#CC1(C(=O)NCC(CC)N2CCCC2)CCN(C(=O)C(C(C)C)SC)CC1 CC1CN(C(c2ccon2)=O)CC2(CCN(C(C3CCC=CCC3)=O)CC2)O1 C(CC1=CCN(C(c2ccc(Cl)s2)=O)CC1)NC(C1OCC(C)C1)=O c1(OC)cc(C)c(NC(C2CC(O)CN2Cc2sccc2Cl)=O)cc1OC N1(C(c2ccc(C#N)cc2)=O)CCc2cc(C(=O)NCC3CCCO3)cnc2C1 CN1CCC(NC(C2(CNC(C3OCCC3(C)C)=O)CCCC2)=O)CC1 N1(C(C2N(C(CC)=O)CCCC2)=O)CCC2C(C1)CN2C(=O)Cc1ncc(C)[nH]1 N1(CC(=O)NCC2CCCNC2)CCc2ccccc2C(O)C1 CCC(CC)(C(=O)N(C1CCN(C(=O)COCC)CC12CC2)C)c1ccccc1 c1(N(CCOC(C)C)C)ccc(NC2(C(N3CCC(OCC)CC3)=O)CC2)nc1 Cc1cn2cccc(C(=O)NC(C)CNC(=O)Cc3ccc4c(c3)OCO4)c2n1 c1(C(=O)NC2C(NC(CC3CCCN(C)C3)=O)C2)ccc2c(c1)OC(F)(F)O2 c1(N(CCCCCC=C)C)[nH]c(=NCC2(NC(C)=O)CCOCC2)nc2sccc12 N1(C(C2(CSC)CCOCC2)=O)CCC2(CC1)CC(N(C(=O)C(C)C(C)C)C)C2 c1(N2C(C)CC(NC(=O)C=C(Cl)Cl)C2)nc(C2CC2)nc2c1CCC2 c1(OC)ccc(CC(C)C(=O)Nc2conc2C)cc1OC CC1(Nc2cccc(OCC(N3CC(S(C)(=O)=O)C3)=O)c2)CCC(=O)CC1 C#Cc1cnc(NC(C2CC23CCN(C(C2CCCC(C)C2)=O)C3)=O)cn1 c1(CC(=O)N(CC(=O)NC(C)C(=O)NC2CC2)CC2CC2)ccn(C)c1 Cc1cc(C2CC2)ncc1C(=O)NC(C)CCNC(=O)Cc1csc(Cl)n1 C1(NC(CS(C)(=O)=O)=O)CC2(C1)CN(C(=O)Cn1nccc1-c1ccccc1)C2 C(CO)(CCCNC(=O)C(C)Cn1ccnc1)NC(C1(C#C)CC1)=O CCCCCC(O)C(=O)N(C1CCN(C(=O)CN(S(C)(=O)=O)C)CC1)CCOC c1(C(=O)NC2CC(O)(CNC(C3CCCC3F)=O)C2)ccc2n[nH]cc2c1 C1(NC(C(CC=C)NC(=O)C=C(C)C(C)C)=O)CC2C=CCC(C1)C2 CCC(C)C(O)CC(=O)N1CC(CCNC(=O)CCC(=O)c2ccccc2N)C1 c1(CN(C)C)ccc(CNCCc2ccccc2I)cc1 C(=O)(CS(=O)c1ccc(Cl)cc1)NC1CN(C(C2CC(C)(O)C2)=O)CC12CC2 c1(C(=O)NC2(CNC(C(CCC)(C)O)=O)CCOC2)ccc(C)c(OC)c1F C1(C(=O)N(CCCNC(C2(C)CCOC2)=O)C)(COC)CCOC1 N12CCC(C1)CC(=O)NCC1CC1CC2=O.C1(C(=O)NC2CC2)(SC)CC1 c1(OCC)ncc(C(N2CC(NC(c3ccoc3)=O)C(O)C2)=O)cn1 C1(C(=O)NC(CCNC(CC(C)C(F)(F)F)=O)C)CCC2(CC1)CC(N(C)C)C2 Cn1nccc1C(C(=O)NC1(CO)CCC1)NC(C1CC1(F)F)=O C(=O)(CCC(C)(C)OC)N(CC(=O)NCC(F)C1CCC1)CC CCCC(C(O)C(=O)N1CC(CO)CC(C)(C)C1)NC(=O)COC C1(C(=O)NC)Cc2ccccc2CN1C(=O)C(=O)NCC1CCC(F)(F)C(=O)N1 N1(C(c2cn(CCC)nc2C)=O)CCN(C(c2cc(C#N)cn2C)=O)C(CC)C1 C(=O)(C(F)CC(C)(C)NC(=O)C(F)n1ccnc1)NC(c1c(C)ncs1)C C1(CC)CN(C(C2COCCN2C(=O)CCn2ccnc2)=O)CC(=O)N1 C(=O)(C(C(C)(C)C)C1CCCCC1)NC(CNC(c1c(C)onc1)=O)(C)CO N1(C(COCCC(C)C)=O)CCOC(CN(C)C(C2(N(C)C)CCC2)=O)C1 c1(CCNC(=O)Nc2sc(C)c(C3CCC3)n2)cc(O)nc(O)n1 c1(CCOCCCC)nc(CCN2CCCC2)nn1-c1cccc(OCC)c1 C1(C(=O)NC(C)C(CO)NC(c2cc(=N)[nH]c(Cl)n2)=O)CC12CCSCC2 C(C)(C)(C(C)CC(=O)N(C(C)CN(C)C(C)=O)C)NC(c1c(C)cc(C)o1)=O C1(C(=O)NCC(CO)NC(C=NOC)=O)CCC(O)(C(F)(F)F)CC1 C12(C(=O)OC)CC(C(=O)N(C3CCC(OC)C3)C)(C1)OC2C C=CC(C)(O)CC(=O)NCC(CC1CC1)C(=O)N(C)C(C1CCOCC1)C N#Cc1csc(CNC(N2CCN(Cc3cccc(I)c3)CC2)=O)c1 C12(C(=O)OC)CC(N)CC1CN(C(=O)COc1nn(C)cc1[N+](=O)[O-])C2 C(C(CC(C)C)NC(=O)C(F)(F)c1cnn(C(C)C)c1)NC(c1ccc(C)s1)=O C(CN=c1nc(N(C)Cc2ccc(Cl)cn2)c2sccc2[nH]1)c1nnc(C)n1C CC1CCNCCC1N(c1cccc(C(C)C)n1)C(C12CC(CO)(C1)C2)=O C(=O)(C#CC(C)(C)O)NC(COC)CC(=O)NCc1nc(C)sc1C C1(CNC(CN(C(=O)C(N2CCOC2=O)C)CC)=O)CCOC1(C)C c1(C(N2CCC(NC(CC3(COC)CC3)=O)CC2)=O)csc2c1C(C)(C)CCC2 C(=O)(CS(=O)(=O)CCO)N1C(CCCNC(C(C)SC(C)C)=O)CCC1 C(=O)(CC1COc2ccccc21)N1CCC(NC(c2c(C)sc(O)n2)=O)C(O)C1 C(=O)(C(C)(C)C(C)NC(C1CCC2CC1CO2)=O)NC(CC)CCO C1(C(N2CC(CNC(CCC=C(C)C)=O)C2)=O)CCCC(N2CCCC2)C1 C1(NC(C(C)(C)NC(C(C)(C)NC(=O)OC)=O)=O)CCCC2(CCC2)C1 C1(CC(=O)Nc2ccon2)(NC(CN(CC(C)(C)C)C)=O)CCC1 c1(C(N2CCC(N(C(c3ccc(C(C)C)o3)=O)C)C2)=O)cc2occc2s1 C1(C(N2CC(C(C)NC(C3(C#N)CCCC3)=O)C2)=O)CCCC(C)CC1 c1(C(=O)NC(C2CCCC2)CNC(C2CC2C(F)(F)F)=O)ncn2c1CCC2 C1(C2(OC)CCC2)(NC(C2N(C(C(C)=CC=C)=O)CC2)=O)CC1 c1(C(=O)NC2CC(N(C(C(C)SCCCC)=O)C)C2)cnn2c1OCC(C)(C)C2 O=C(C1=CS(=O)(=O)c2ccccc21)NCC1CCCC(CNC(C2(O)CC2)=O)C1 C1(NC(COc2ccc(SC)cc2)=O)CC2CN(C(C3CCCN(C)C3)=O)CC12 c1(C(C)NC(C2CCOC2CNC(=O)C(=O)NC2CC2)=O)cncc(F)c1 CC1CC2(C(=O)N(C3CCCC3)CCNC(=O)C=CC3CCOC3)CC12 N12CCC(C1C1CC1)NC(=O)C1(C3CCC13)C2=O.c1(C=O)ccco1.CO N1(C(C2N(C(c3ccc(C#C)nc3)=O)CC(F)(F)C2)=O)CC2(CCOC(=O)N2)C1 c1(Cc2nnc(N3CC=CC(OC)C3)n2CC(C)CN(C)C)ccc(C)c(Br)c1 CC#CCCC(=O)NC1CCCCC1NC(c1c(O)noc1C)=O C1(NC(Cc2cn(C(C)C)nc2)=O)CN(C(=O)CCn2ccnc2)CCC1CO c1(C(=O)NC2C(CNC(c3cnn(C)c3Cl)=O)C2)cc(Cl)cc(F)c1N c1(OC)cc(Br)ccc1CC(=O)NC1CC(C(=O)NC2CONC2=O)C1 c1(OCC(=O)NC(C)CC(C)NC(c2cc(C(N)=O)c[nH]2)=O)ccccc1C#N O=C1CN(C(=O)C2=CS(=O)CCC2)C2CCN(C(=O)Cc3c[nH]nc3O)CC2N1 C1(C(C)NC(=O)C(O)C2CCCC2)CCCN1C(=O)CC1(N(C)C)COC1 CCCC(CNC(c1cncs1)=O)C(=O)NCC1(O)CC(O)C1 C1(C(=O)Nc2sc(-c3ccccc3)nc2Cl)CNCCN1Cc1ccc(Br)cc1 CCC(C(=O)N1CC2CC(C1)CN(C(C1CC3(C1)CC3F)=O)C2)C(C)(C)CC c1(C(=O)NC(C2N(C(C3(OC(C)=O)CC3)=O)CCC2)C)ccncc1Br C(=O)(C1CCCc2sccc21)N1CC(C)CN(C(c2ccnc(C)n2)=O)C(C)C1 C(=O)(CC#Cc1ccccc1)NCC1C(C)(C)CC1O N1(C(CC2C=NN(C)C2=O)=O)CCCC(C2(NC(=O)Cc3cccnc3)CC2)C1 C1(CCCC)CN(C(c2cc3n(n2)CCC3)=O)CCN1C(c1cnc(C)nc1)=O C1(CC=C)(NC(C2CCOC2)=O)CCCN(C(=O)CC=CC)C1 C(C(CC(C)C)C(=O)NC1CN(C(c2ccc(C)s2)=O)CC12CC2)OC N1(C(c2c(C)con2)=O)CC(C)C(NC(C2CCC(CC#N)CC2)=O)C(C)C1 n1(CCC)ncc(C(=O)NC(CNC(C2CCCS2(=O)=O)=O)C(C)(C)C)c1Cl CC(F)(F)C(F)(F)CC(=O)NC1CCC1NC(C1C2C3CCC(C3)C12)=O CC1(C)CCC(CCNC2CC3CC3(COC)C2)CC1 C(C(C(C)C(C)C)NC(c1nsnc1O)=O)NC(c1ccc(C)cc1)=O C1(OC)(CNC(=O)C(O)CN(C)C)CCN(C(=O)CSCc2ccc(Cl)s2)C1 C#CCCCCC(=O)NCC1CCC(NC(C2(O)CCCC2)=O)C1 CCC(C(=O)NC1CCC(CC(=O)N(CC(C)OC)C)C1)C(F)(F)F c1(C(N(CCNC(C2CCN(C(C(C)C)=O)CC2)=O)C)=O)ccc(O)c(F)c1F c1(OC)cc2c(cn1)N(C(=O)CSc1c(C)oc(C)c1C)CC2 N1(C(=O)OC)CCCC(N=c2nc3c(ncn3C)c(NCc3cc(Cl)no3)[nH]2)C1 c1(CCNC(C(c2ccc(Cl)cc2)(C)O)=O)ncc(Br)cn1 N1(C(CCC=CC(C)C)=O)CCN(C(=O)C2=CCCCC2)CC1CC1CC1 C(=O)(C#CC1CCCC1)NC(C(=O)NCc1scc(C)n1)CC(N)=O c1(COC)cc2ncc(-c3ccc(C#N)c(OC(F)(F)F)c3)cc2[nH]1 C(CCCC(=O)NCC12CC1CN(C(c1cccn1C1CCCC1)=O)C2)N(C)C CC1CCCC(C)N1CCC(N1CCOCC(NC(=O)Cc2cnoc2)C1)=O N1(C(CC(C)C(F)F)=O)CC2CCC1C(CNC(C1CCC(F)(F)C1)=O)C2 C[S+](C)CCC(O)C(=O)NCC1C=CCN1C(c1cc(C(N)=O)no1)=O Cc1cccc(-c2cccc(Nc3nccc(N4CC(CO)C5(CC5)C4)n3)c2)c1 c1(C(=O)NC2CC(CCNC(=O)CNc3ncccn3)C2)ccc(F)c(O)c1 C1(CC)CN(C(c2cnccn2)=O)CCC1NC(c1cc(O)nc(O)n1)=O N(C(=NCC1CCOC1)NCC1C(C)(C)C1(C)C)CC(c1ncccc1F)(C)C c1(N(C)CCSc2ccccc2)nc(=N)nc(N2CC3CCC3(C(F)(F)F)C2)[nH]1 c1(C(=O)NC2(C(N3CCCC(OC)C3)=O)CCN(C)C2)cc2occc2[nH]1 CN1N=C(C(=O)N2CCCC(O)(CNC(=O)CCCC(F)(F)CO)C2)CCC1=O c1(C(=O)NC2CCCC(NC(C#C)=O)C2)c(Cl)cccc1[N+](=O)[O-] N1(C(c2c(C)nn(-c3cccc(Cl)c3)n2)=O)CC(NC(=O)CC2CC2)CC(O)C1 CC1CC(C(=O)NCC(C)(C)CCNC(c2cc(C3CC3)on2)=O)CCS1 Cc1cc(C(=O)NCCOCCNC(=O)C(O)C(C)(C)C)cc2c1CCC2 C1(CNC(c2c(C)occ2)=O)CCCC12CCN(C(C1(C(C)C)COC1)=O)CC2 c1(C(=O)NCC2CCCCC2NC(c2sccc2Cl)=O)occ2c1CCOC2 C1(NC(CCCC#C)=O)CC2CCC1N(C(=O)CCc1cnoc1)C2 c1(NC(C)=O)cc(C(=O)N(CCCNC(=O)C(F)(F)C(C)O)C2CC2)ccc1C c1(C(=O)OC)cc(=NCCN(C(=O)CC2CCN(C)C2=O)C)[nH]cc1[N+](=O)[O-] O=C(C1=CCC(NC(=O)CC2COC(=O)C2)C1)NCCCC1CCCCO1 Cn1ccc(C(=O)NCC2COC(CNC(=O)CC3(N4CCCC4)CC3)C2)n1 CC1(C2CC2C(=O)NC2CCC(CC(=O)NCc3ncc(F)cn3)CC2)COC1 CCC(C)CCCCC(=O)NC1C2CCN(C(=O)C=C(C)C(C)(C)C)C12 C=CCCCCCCC(=O)N(C1CN(C(=O)C(C2CCOCC2)C)CC1(C)C)C C1(CC(=O)NCCCOC)CCCCN1C(C1CN(S(=O)(=O)C(F)(F)F)C1)=O C(CCC(=O)NCC1(CNC(=O)COC)CCC1)NS(C)(=O)=O.C1(C)CC1(F)F C1(C(=O)OC)CCN(C(=O)C2C=CCN(C(=O)CCc3nc(=N)[nH][nH]3)C2)O1 N1(C(CCN(CC)CC)=O)CCC(C(N2CCC2(C)C(=O)OC2CC2)=O)C12CC2 Cc1cc(OCCC(=O)NCC2CCN2C(C2COC(=O)O2)=O)cc(C)c1 C=C=CC(C)C(=O)NC(C1(C(=O)NC(C)CO)CC1)C c1(CNC(CN(C(C)C)C(C2CCC2C(C)(C)C)=O)=O)ccncn1 C1(NC(CC(CC)O)=O)CC2CCC(C1)N2C(=O)C(C)Cc1ccccc1C C#CC1(C(N2CCC(NC(c3cc[nH]c(=N)n3)=O)C2)=O)CCCC1 Cc1nc(NCC2CCC(NC(C3CSCCS3)=O)C2)c2cnn(C)c2n1 c1(C(N(C2CCCC(NC(CC(C)C)=O)C2)C)=O)ccn(C)c(=O)c1 C1(NC(CN2CCN(C(C(COC)(C)C)=O)CC2)=O)COCC(C)(C)C1 C1(OC)CN(C(=O)C(c2cccnc2)O)CC1C(N1CCC(N2CC(O)C2)C1)=O C1(CNC(Cn2c(C)ncc2)=O)CCC12CCN(C(=O)C(C1CC1)C1CC1)CC2 c1(C(CC)NC(N2CCCC(NC)CC2)=O)nc2ccccc2[nH]1 N1(C(COC(C)=O)=O)CC2(C)CN(C(c3ccc4nnc(O)n4c3)=O)CC2(C)C1 n1(CC)ncc2c1CC(C(=O)NCC1CN(C(=O)Cc3cn[nH]c3)CC1O)CC2 c1(C(N2C(CN(C(c3cnc(SC)s3)=O)C)COCC2)=O)cc(Cl)ncc1N CC1C(NC(c2ccncc2C2CC2)=O)CC2CCC1N2C(=O)CC1CC1(Cl)Cl CCCCCCCC(=O)N1CC2CC2C1C(=O)NCCN1CCC1 c1(C(=O)NC2(CNC(CC3CCC(C)(C)O3)=O)CCCC2)cnc2[nH]cnc2c1 Cc1nc(N(C)CC2CCN(C(C3CN(CC(F)(F)F)C3)=O)C2)c(C)c(C)n1 Cc1cc(C(N2CCSC(C(=O)Nc3ccc(F)cc3Cl)C2)=O)cnc1F c1(C(N2CC(NC(C3C(C(=O)OC)C3(C)C)=O)C2)=O)cn(C)nc1C CN1CCN(C(c2ccccc2CN(C)C)=O)C(NC(=O)CN2CCCCC2)C1 C1(F)(C(=O)NC(c2ncnn2C)CC)CCCN(C(=O)C2=C(C)CC2)C1 CCC(CC(=O)NCC(F)CNC(=O)CC1CCOCC1)C(C)C C(=O)(C#CC(C)(C)C)N1CCC(CC)C1CNC(c1ncn2c1CCC2)=O N1(C(COC)=O)CCC(CN(C(C2NC3CCC2C3)=O)C2CC2)CC1 N1(C(c2cc(CCOC)on2)=O)CCCCC1CC(C)NC(=O)C(Cl)=CCl C1(C(C(=O)NCCCC)N(CC)Cc2ccc(C)cc2)CCOC1(C)C C1(NC(C2CCc3c[nH]nc3C2)=O)CC2CN(C(=O)Cn3cc(Cl)cn3)CC2C1 C1(C(=O)NCCC(C)O)(CO)CCN(C(=O)CCc2ncccn2)C1 c1(C(=O)NCC2(CNC(C=CSC)=O)CCC2)cnc2cc(O)ccc2c1 C1(NC(c2c(C)cc(N)cc2)=O)CCN(C(C2C(C)C2C)=O)CC12CCC2 CCC(C)(C)C(O)C(=O)NCCC1=CCN(C(=O)CCC2CCC(=O)NC2)CC1 C1(NC(CSCC(C)C)=O)CN(C(c2cnn(C3CCCCC3)c2)=O)CC1(C)C c1(C(=O)NCC(C)CNC(C2(C)COCCO2)=O)ccc2c(ccn2C)c1 c1(CC)ccnc(C(=O)NC2CCCC2C(=O)NC(c2scnc2C)C)c1 CN1C(=O)Cc2ccc(C(N3CCC(NC(=O)CS(N)(=O)=O)C(O)C3)=O)cc21 CC1C2CCC(C2)C1C(=O)NCC(O)CC(=O)N(C)Cc1cccnc1O CC1(C(=O)NC23CCC(CC2NC(C24CC(F)(C2)C4)=O)C3)CCCCNC1=O CCC1=NOC(CC(=O)NCCCNC(c2ccncn2)=O)C1 c1(C(=O)NC(CC)(C)CNC(C2CCCCN2C)=O)cc2cccc(OC)c2o1 CC(=O)CCCCC(=O)NCC(O)CC(=O)NCC(C)(C)C1CCCO1 N1(C(C(=O)NCCc2cnc(C)s2)=O)CCCCCCC1C C1(NC(C(CC)(C)O)=O)CC12CCN(C1CC1CC(C)(C)C)CC2 C1(CCC)CN(C(c2ccc(N)c(F)n2)=O)CCN1C(c1nocc1C)=O C12(C(=O)NCC3(OC)CN(C)C3)CC(C)(CN1C(C1CCC(C3CC3)O1)=O)C2 C1(C(C(=O)NCCN(C(Cn2c(CCC)ncc2)=O)CC)C)CCC(C)(C)CC1 C1(C(=O)NC(CC=C)CNC(c2ccon2)=O)CCCCN1C(C)=O C1(CC(=O)NCCOCC(=O)NCC2CC2CO)CCCCCC1 CC1(C)CCN(C(C2CC(=O)NC(=O)N2)=O)C1CC(=O)NCCc1nncs1 N1(C(C=CC=CCC)=O)CCCC(C)C1CNC(c1cn(C)nc1CC(C)C)=O N1(C(C2CC(OC)C2)=O)CCC(N(C(=O)CCOC2CCC2)CCO)CC1(C)C S(=O)(=O)(c1ccc(N(C)CCc2cncs2)c(Br)c1)N(C)CC1CCCN1C Cc1c(C(N2CCCC(NC(C3(C)CCCN3C)=O)C2C)=O)cnc2ncnn12 c1(C(=O)NCC(CC)NC(c2cccc(C)c2)=O)nc2n(c1C(C)C)CCCC2 CC1CCN(C(C2CC(O)C2)=O)CC1CNC(c1cccc(C(N)=O)n1)=O C1(CCNC(C2C(C(=O)OCC)C2)=O)CN(C(=O)CCOC)CC1C c1(COC)nnc(SCC(=O)NC(=O)NC)s1 c1(C(N(CC(C)(C)NC(C2CC2C(F)F)=O)C)=O)cn(C2CCOC2)nn1 Cc1cc(CCNC(C2(CO)CCN(C(=O)CCN=[N+]=[N-])C2)=O)nn1C N1(CC)C(=O)CCC1C(=O)NC1CCC1NC(c1ccc(C)nc1)=O N1(C(CCN(C(=O)C(n2ccc(C)n2)C)CC)=O)CCCN(C)CC1C N1(C(Cc2c(C)non2)=O)CCCC2(CC(NC(C3CN(S(C)(=O)=O)C3)=O)C2)C1 N1(C(c2ccn(CC)c(=O)c2)=O)CCC(CNC(=O)CCOC(C)C)C(F)(F)C1 N1(CC(=O)N(c2nnn(C)n2)C(=O)Cn2c(O)nnc2O)CC2CCOC2C1 C=CC(CC)C(=O)NC1(CF)CN(C(=O)C(C)=C2CC2)C1 c1(-n2cc(C(N3CCNC3=O)(C)C)nn2)noc2ccc(F)cc12 N1(C(c2cc(OC)c(Br)nc2)=O)CCC2CN(C(=O)C(C)n3cccc3)CC12 C(=O)(C(C)C(F)(F)F)N(C1CCN(C(C2(F)CCC2)=O)CC1)CC#C N1(C(CC2C(C)CCO2)=O)CCC2(C1)CN(C(=O)CCC1(C)CCC(=O)N1)C2 CN=c1cc(C(=O)NC2(C)CN(C(=O)Cc3cccnc3)C2)c(Br)c[nH]1 c1(C(N2CC(N3CCN(C(C4OCCO4)=O)CC3)C2)=O)c(F)cccc1Br C(=O)(C(C)(F)C(C)(C)F)N1CCCC(CN(C(C(CCC)NC(N)=O)=O)CC)C1 CC1CCN(CC(=O)NC(C(=O)NCCCS(C)(=O)=O)C2CC2)CC1 Cc1cc(F)c(C(N2CCOC(C(C)NC(=O)CCCC(F)F)C2)=O)c(Cl)c1 C1(C2CC2)(CNC(c2ncc(C)c(Cl)c2)=O)CCN(C(=O)CCCC2CC2)C1 C(=O)(C(C)CC#N)N1CC(C(N(CC=C)CCO)=O)(CC=C)C1 Nc1cc(C(N2CCC(O)(CNC(C3CC4CC34)=O)C2)=O)c2c(c1)OCCO2 C1(CN(C(=O)C(N2CCCC2c2ccc(Cl)cc2Cl)=O)C)CCC2(CCOCC2)C1 c1(OC)cccc(N2CCN(C(C3(c4ccccc4)CCNCC3)=O)CC2)c1 CCCC(CC(=O)OC)NC(=O)NCCCN1C(C)CCCC1C C1(NC(CC2C(NC(C3(CN(C)C)CC3)=O)CCC2)=O)C2CCCOC12 CC(CS(C)(=O)=O)C(=O)NC1CCN(c2nc(C(F)F)nc(=N)[nH]2)C12CCC2 N1(C(c2cn(C)nn2)C(=O)NCCCC)CCCC(C)C1C(=O)OC Cc1nc(N2CC(CNC(C3CCCOCC3)=O)CC2C)cc(C(F)(F)F)n1 c1(C(=O)NC(C(C)(C)NC(c2ncnc(C)c2C)=O)C)cccc2cnccc12 CC(C)CC(C(=O)NC1CCC(=O)NC1)ONC(=O)CN1CCSCC1 N1(C(CC2(C#N)CCC2)=O)C2CCC1C(C(N1CCCCC1C1CCC1)=O)C2 c1(CC)ccc2cc(C(=O)NC34CC(C3)N(C(C3(F)CCOCC3)=O)C4)[nH]c2c1 C(CCCCC(=O)NCc1cccc(OC)c1)N(C(C(C=C=C)C)=O)C C1(NC(c2c(C)ncnc2)=O)CCN(C(c2sccc2F)=O)CC1C(C)C C#Cc1cccc(CC(=O)NC(CCF)C(=O)NCCCOCC)c1 C=CCC(CC(F)F)C(=O)N1CCN(C(=O)C(C)n2cncn2)C2(CCC2)C1 c1(NC(C(C)N(CCC)C(c2ncccn2)=O)=O)cccc(F)c1O C1(CNC(CC(n2ccc(C)n2)C)=O)CC(C)N(C(=O)C(C)c2ccco2)C1 S(=O)(=O)(c1cnc(N2CCC3(CCSC3)C2)c(Cl)c1)NCc1c(=N)cc[nH]c1 c1(C(=O)NC2C(NC(c3[nH]nnc3C3CC3)=O)CCCC2)cccc2cc[nH]c12 c1(N2C(C)CC(CNC(c3ccc(SC)cc3)=O)C2)cc(=O)n(C)c(=O)n1C N1(C(C2CC(C)(CC)C2)=O)CCC(Nc2cc(C)ncn2)CC1 c1(C(=O)NCC(C2CCC2)NC(C2CCCOCC2)=O)ccn2c1CCCC2 C1(C)(CC(=O)OC)CCN(C(=O)NC(c2ccc(Cl)c(Br)c2)C)CC1 CON=C(C(=O)NC(C1CN(C(c2cc(C)c(C)o2)=O)C1)C)c1ccco1 N1(C(C(C)NC(C=C(CC)C)=O)=O)C(C)CC2CN(C(C3OCCC3CC)=O)CC12 c1(C(C)=O)cccc(CN(C(=O)COC2(C)CCC2)C)n1 C(C(=O)NCCN(C(=O)CC1CC1)C)(c1cccs1)NC(=O)O.C(C)(C)(C)OCC#N C1(C)(C(=O)NCC(C(=O)NCCN(CCOC)C)OC)CC(=O)N(C)C1 C1(CNC(C2N(C(=O)C(C3(O)CCCC3)F)CC2)=O)(CO)CCCCO1 C(=O)(CC(O)C(C)C)N1CCC(F)(CNC(C2CC(CC)C2)=O)C1 C1(NC(c2occ(C)c2C)=O)CCN(C(=O)C(F)(F)N2CCOCC2)CC1CO c1(C(=O)NC23C(CN(C(c4cnc(OCC)nc4)=O)C2)C3)ccc2cc[nH]c2n1 N1(c2snc(C(=O)OC)n2)CCCC2CN(C(=O)CCC3CC3(C)C)CCC12 c1(COCCOCCOC)cc(NC(C2CC(O)C2)=O)ccc1Cl Cc1cnc(C(=O)NCC(C2CC2)N(C)C(C2(C)CCNC(=O)C2)=O)cc1C N1(C(C(C)c2cc[nH]n2)=O)CCC2(C1)CN(C(=O)CCC(F)(F)F)CCO2 C1(NC(c2cnc(C)o2)=O)CCC2CN(C(C3CCSCC3)=O)CC2C1 N1(C(C2(CNC(C34CCC(C3)C4)=O)CC2)=O)CCC(C(C)(C)OC(C)C)CC1 c1(CC)cccc(C(=O)N(C)CC2CCN(C(=O)C=NOC)C2)c1 CC1CCCC(OCC(=O)NCCNC(C2CC(O)(c3ccccn3)C2)=O)C1 C=CC1CCCCN1C(C1CC(F)CN1C(c1ccc(F)cc1C)=O)=O C(=O)(N=S1(=O)CCC2(C1)NC(=O)NC2=O)c1ccc(CN(C(C)=O)C)cc1 c1(C(=O)N(C(Cc2cnc[nH]2)C(=O)N2CCC2C2CCC2)CCO)ccc(O)nc1 CCC1=C(C(=O)NC2CCCC2CNC(c2cc(C)c(F)cc2F)=O)CCCO1 C1(C(=O)NC23CCCC2CN(C(c2ccc(F)o2)=O)C3)CCc2nnc(O)n2C1 N1(C(C2(C(=O)OCC)CCCCO2)=O)CC2CCC(C1)N2C(=O)CC(C)COC C(=O)(C#CC1(C)COC1)NCC1(O)CN(C(c2c(C)ccc(C)n2)=O)C1 c1(C(=O)NCC2C3CN(C(C4(C=C)CCOCC4)=O)C2C3)cnc2[nH]ccc2n1 c1(C(N2CCN(CC(=O)OC)CC2)=O)cnc2n1CCOC2 Cc1ccc(C(C)NC(=O)CC2CCCN2C(c2coc(C)c2)=O)nc1 C1(NC(c2c(COC)ncs2)=O)CCCCCC1NC(c1oncc1C)=O CCCC(C)(O)C(=O)NCC1CC2(CC(NC(c3cc(C4CC4)nn3C)=O)C2)C1 Cc1cc(NC2CCN(C(c3nc4ncccn4n3)=O)C2)n2nc(C)nc2n1 N1(C(Cn2c(C(=O)OC)cnc2)=O)CCCC2(CNC(=O)C2)C1 c1(NC(N)=O)ccc(C#N)cc1[N+](=O)[O-].CC(C)CC1CNC(C(C)C)C(=O)N1 c1(OC)ncc(F)cc1C(=O)NCC1CCCCN(C(=O)Cn2cnnc2)C1 N(C(=NCCc1ccccc1)N1CCC(Br)=C(C)C1)Cc1ccc(N(C)C)cn1 C(=O)(C(C)(C)C1=CCN(C(c2cc(COC)on2)=O)C1)N1C(C#C)CC1 c1(CC)c(C(=O)N(CC(C)O)CCNC(=O)CC2(C)CC2)cnn1C C12(NC(CN(S(N(C)C)(=O)=O)C)=O)CCCC1CN(C(C1CC3CC3C1)=O)C2 CC1(C)CCCN(C(=O)C=CC=C(Cl)Cl)C1CNC(C1CC12CCCC2)=O c1(C(N2CCC(OCCCNC(CCSC)=O)CC2)=O)cncc(P(C)(C)=O)c1 n1(CCOC)cc(CNC(C2(C)CCOCC2)c2nnnn2C)c(C)n1 C12(NC(CC(C)(C)SC)=O)CCCC1(F)CN(C(C1(C)CC(C3CC3)=NO1)=O)C2 c1(CCC(=O)NC(CCNC(c2nc(C)nn2C)=O)(C)C)cnc2ccccn12 C1(C(=O)NCCC2(NC(CCCCCCC)=O)CCC2)CN2CCCCC2CO1 Cc1cc(=NC(=O)CC(O)c2ccccc2)[nH]n1-c1ccc(Cl)c(Cl)c1 Cn1ncc(C#N)c1NC(c1ncc(-c2cnoc2)cn1)=O c1(OC)nc(C(=O)N(C)CC2(C)CCCC2NC(=O)Cc2cccnc2)sc1C C1(NC(=O)CNC(C2CCOCC2)=O)CC2CC(C1)N(C(C1CCCCO1)=O)C2 c1(NC(N(c2nccc(OC)n2)C2CCCNCC2)=O)cccc(Cl)c1F C(C(F)(CO)c1ccccc1)N(C(C(N1CCOCC1)C)=O)c1nccs1 C(=O)(C(C)CC(C)(F)F)NCC(CC)NC(c1ccc(Br)c(N)c1)=O C(=O)(C1(C)COc2ccccc21)NCC1C(C)(C)CCN(C(C2(O)CCC2)=O)C1 S(=O)(=O)(c1ccc(C#N)cc1)NC1CCCN(C(=O)OC(C)(C)C)C1 CCCCC(O)C(=O)N1CC(C)(OCC(=O)N(C(C)C(=O)OC)CC)C1 C=C(C)C(O)CC(=O)NC1(CNC(c2nc(CC(F)(F)F)sc2C)=O)CC1 Cc1cc(CNC(=O)CC2(C)CN(C(=O)NC3CCCCCC3)C2)cc(Br)c1 C1(NC(C(Cc2cn[nH]c2)NC(=O)CC2CNC(=O)O2)=O)CCC2(CCCC2)C1 C1(C(=O)NCCC(=C)C)CCCCCC1NC(c1cc(C(C)C)[nH]n1)=O C1(CNC(C2C(C=C)OCC2)=O)CC2(C1)CN(C(=O)C(C)NC(C1CCC1)=O)C2 C12(CNC(C3CCN(C(CN(C(C)C)C(C)=O)C)CC3)=O)CCCC1OCC2 N1(C(C2CCCN2C)C)CCCCCC1C=Cc1cccs1 C(=O)(CC(C)(O)C(F)(F)F)NCC(C(C)(C)C)NC(c1c(C)ccc(Cl)c1)=O CC1CCC(Cl)=C(C(=O)NCC(C)NC(=O)CCN2CCCC2)C1 c1(C(c2ccccn2)(n2nccn2)C)nc(-c2cccs2)nn1CCn1ccnc1 c1(C(c2ncnn2C(C)C)NC(C=C)COC)nnnn1CC N1(C(C(C)NC(C)=O)=O)CCC2(CCC(NC(C3CN4CCN3CC4)=O)CC2)C1 CCC(C)(O)C(=O)N1CCC(O)(CNC(=O)CCCc2cncs2)C1 CCCCCCCCC(C)C(=O)N1CCN(C(=O)C2=CCOC2)CC1C1CC1 CN1CC(C(N2CCN(C(c3ncccc3C(F)F)=O)CC2)=O)CC1=O c1(CN2CC(CCNC(C)=O)(NC(C)=O)C2)ncccc1Cl CC(C)CC(C)C(=O)N1CCOCC1CN(C)C(c1cc(F)c[nH]1)=O O=C1NCC2(CN(C(=O)CC3CCN3C(=O)C(C3(O)CCCC3)F)C2)N1 C(=O)(C(C)(C)CC1CC1)NCC(CCNC(CN(C)C(=O)OC(C)(C)C)=O)O C1(C(C)NC(=O)Cc2csc(Br)c2)CCN(C(=O)C=CCF)CC1 c1(C(c2ccncc2)NC(=O)CC2COC(=O)C2)ccc(F)cc1 Cc1ccc(Cl)c(F)c1C(N1CCC1CNC(C1CCC2CC12)=O)=O c1(NC(C(C)N(CCC)C(C2CC(O)C(F)C2)=O)=O)cc(C)c(F)cc1C c1(OC)ccc(C)c(OC)c1C(=O)NCC1CC(F)CN1C(=O)C1=CC(C)(C)C1 CC1CCN(CC(=O)NCC2(O)CN(Cc3cccc(Cl)c3)C2)CC1 O=C1NCC2(CCCN(C(C3CCCN(C(c4cc(Br)ccn4)=O)C3)=O)CC2)N1 C1(C(=O)NCCC(CNC(CC2(COC)CC2)=O)(C)C)CCn2ncnc2C1 C1(CNCc2c(-c3ccc(F)cc3)n[nH]c2)COC2CCCC2O1 c1(C(=O)NC(C2CCCN2C(=O)CCC2CCCOC2)(C)C)n[nH]cc1Br N1(C(CCCN(C)C)=O)CC2C3CCC(C2C1)N(C(c1cnc(O)s1)=O)C3 N1(C(c2on(C)c(=O)c2)=O)CC(NC(c2cnn(CCO)c2)=O)CC12CCC2 c1(C(N2CCC(O)(CCNC(C(C)C(C)O)=O)C2)=O)c(N)cccc1F C(=O)(C(C1=C(C)C=CCC1(C)C)N(Cc1ccccc1C)CC1CC1)NCC=C N1(C(c2c(C(=O)OC)cco2)=O)CC(NC(=O)C(c2ccccc2)O)CCC1C c1(C(N2CC(=O)NCC2)=O)cc(I)ccc1N1CCCC1.c12ccc(cc1)CO2 C(=O)(N=c1ccn(C2CC2)[nH]1)C1C(c2cn(C)nc2)N(C(C)(C)C)C(=O)C1 N1(C(C2N(C(C)C)CCC2)=O)CCC(O)C(C(N2CCC2CO)=O)C1 c1(C(C)C)cc(NC2(C3CN(C(=O)CCc4cc[nH]n4)C3)CC2)n2ncnc2n1 c1(C(=O)NC(CCC#C)C(=O)NCCc2cn(CC)nn2)n[nH]c2ccccc12 c1(OC)c(CN2CCOC(COC)C2c2ccnn2C)cc(C)cc1C C1(CNC(c2occ(C(C)(C)C)c2)c2nnnn2C(C2CC2)C2CC2)CCCNC1=O C(CN=C(NCc1ccccc1Cl)NCc1cncn1C)OCC c1(OC)cc(NC(C2CC(NC(c3coc4ccccc34)=O)C2)=O)c(Br)cc1Cl C1(NC(C#CC(C)(C)C)=O)C2CC3CN(C(c4ccc5c(c4)CCO5)=O)C1C3C2 O=S1(=O)CC2CC(NC(=NCCF)NCC3(CC4CC4)CC3)CC2C1 CCCCC(C(=O)NC1CCC(F)(CNC(c2csc(C)n2)=O)C1)C(C)C C(CCC(N)=O)(C(=O)N1CCC1(C)CC(C)C)n1cc(C(C)NC)nn1.C1CO1 N1(C(c2n(C)nc(O)c2)=O)CC2OCCN(C(=O)C3=CS(=O)(=O)CCC3)C2C1 C1(C(=O)NCC2(F)CC(CNC(c3ccc(Br)o3)=O)C2)CCCCNC1=O N1(C(c2cc(OCC)n[nH]2)=O)CC(CCNC(=O)COCCF)C(C)C1 c1(CC)ncc2c(n1)CCC(C(=O)NCC1CN(C(C3CC(O)C3)=O)CCO1)C2 N1(C(C(CNC(C2C(CC)OCC2)=O)CC(C)C)=O)CCC2(COC(=O)N2)C1 c1(C(=O)NCCC(C)N(C)C(c2occc2F)=O)cccc2ncnc(O)c12 n1(CC(=O)N(CC(C)O)CCNC(=O)CS(=O)(=O)N(C)C)cnc([N+](=O)[O-])n1 CCC(C)C(C(=O)NCCn1cc(CO)nn1)N(C)C(c1ccoc1)=O CC(C)(C)S(=O)(=O)CC(=O)N1CCC2CN(C(c3ccc(F)cc3F)=O)C2C1 N1(C(Cc2cc(C)ns2)=O)CCC(C2CCN(C(C34CCCC3C4)=O)CC2)CC1 N1(CC(N2C3CN(C(C4CC(C)OC(C)C4)=O)C(C3)C2)=O)CCc2sccc2C1 c1(C(=O)NNC(=O)CSc2ccc(Br)cc2)ccc(Br)c(Cl)c1F CCCCCC(=O)N(C)CCN(C)C(C1CC1c1cnn(C(C)C)c1)=O C1(C(=O)NC(C#CC)(C)C)CCCCN(C(=O)CCc2ccco2)C1 CCC(CC)CCC(=O)NCC(O)CCNC(c1cc(C#N)ccc1N)=O S(=O)(=O)(c1ccc2c(c1)OCCO2)N1CCCC(C(=O)OC(COC)C)C1 c1(C(=O)OC)cc(NC(C2CC2NCc2ccc(C)nc2)=O)cc(C#N)c1 C12(CNC(COC(C)C)=O)CCC(CC1)N(C(=O)CC1CCCNC1=O)C2 C(=O)(C1=CCC(C)CC1)NCC1(OC)CCN(C(=O)Cn2nc(C)cc2C)CC1 C1(COC)CCN(C(=O)CC2(N(C(=O)C(F)=C(C)C)C)CC2)CC1 C1(N2CC(=O)NC2)COC2(CCN(S(=O)(=O)c3cc(C(=O)O)ccc3F)CC2)C1 c1(C(=O)NCCCC(C)(C)NC(c2c(CC)c[nH]c2)=O)cc(F)ccc1C C1(C(N(CCCNC(=O)C=Cc2cccs2)C2CC2)=O)CCc2nnnn2CC1 C1(C)(C(N(C(C(=O)NCCC(COC)O)C)C2CC2)=O)CCCN1C C1(C(N(C(c2cccnc2)C)CC)=O)CC=CCC1C c1(C(=O)NCC(CC)NC(c2ccnn2CC#N)=O)cnc2onc(C)c2c1 C(=O)(C(C)(C)CC(F)F)NC1CC(C)N(C(C2CCC(C(C)(C)C)CC2)=O)CC1 C(CCCC(=O)NC(CC1CC1)C(=O)NCC1(CO)CC(C)C1)OC C1(NC(=O)COCC(F)(F)F)CCCN(C(C2(F)CCOCC2)=O)C1 C1(NC(c2sccc2Cl)=O)CC2(C(=O)NCc3ccc(O)nc3)COC1C2 CCC(C(=O)N(CCC(N1CC=CC1CN(C)C)=O)C)C(C)(C)CC N1(C(C(CC=CC)C)=O)CCCCC(C2CN(C(=O)C(C)(C)CCOC)C2)C1 CS(=O)(=O)C1(C(=O)NCC2C=CCN2C(=O)C=CC=Cc2ccccc2)CC1 CCC(C(=O)NC1CC2(C1)CN(C(=O)C(=O)Nc1cc(F)ccc1C)C2)C(C)C C(=O)(CC(C)N(C(=O)CNC(=O)C(C)C)C)OC(C=CC(=O)OC)C c1(C(=O)NC(C2CCCCC2)C(=O)NCc2cnsc2)cc(F)ccc1O CN=c1[nH]cc(C(=O)NCC2(C(F)F)CCN(C(=O)C(CSC)OC)C2)s1 CN1CCC(CO)(CNC(=O)C(c2cccs2)NC(c2cncnc2)=O)C1 N1(C(Cc2cn(CC)nn2)=O)CC2(CCC(CNC(=O)C(C)c3cccs3)O2)C1 c1(C(N2C(C(=O)OCC)(CNC(C=COCC)=O)CCC2)=O)ccc(C)c(Cl)c1F C1(C2CCN(C(c3cscn3)=O)C2)(NC(c2c(C)cc(C)s2)=O)CC1 c1(NCC)ccc(CNC(=NCC2CCCO2)NCC2(SC)CCCSC2)cc1 CC1(CO)CN(C(C2CC(NC(=O)CCc3cncnc3)C2)=O)CCC1O C1(C(F)(F)F)(NC(C(c2n(C)ncc2)N)=O)CCCN(CCC#N)C1 Cc1oc(C#N)cc1C(=O)NC1CCN(C(=O)CN(C)C)C(C2CC2)C1 C1(C(N(CCCOCCN(C(=O)Cn2cccn2)C)C)=O)CCC12CCCO2 N1(C(C2C(NC(CCCCCC)=O)CCOC2)=O)CC2(CCC(=O)NC2)C1 c1(C(=O)NC(CN(C(C(=O)NC)=O)C)C(C)C)ccc2nc(C3CC3)[nH]c2c1 C1(C(=O)NCC(CC)NC(C2(CC)CCC2)=O)COCCOC1 N1(c2ccc(C(=O)OCC)cn2)CCC(C)C(NC(=O)C(c2cccnc2)C)C1 c1(C(=O)NC(CCCC)CNC(c2cc(C)oc2C)=O)c(C)nc2sccn12 Cc1cn(C(C)C)cc1C(=O)NC1CC(CNC(=O)CCN2CCCCC2C)C1 N1(C(CCC)=O)CCOCC1C(C1CCN(C(c2oncc2C)=O)CC1)(C)O Cc1nn2c(c1CNC(=O)CCCn1cncn1)CN(C(=O)C(O)C(C)C)CC2 N1(C(C2(C(=O)OCC)CC2)=O)CCC2(CC1)CN(C(c1ccc(Cl)cc1O)=O)C2 C(C)(C)(CCCCNC(=O)CCC1CCCCC1)NC(C(CSC)O)=O C=CCC(C)(C)CC(=O)NC(C)(C)CN1CCN(C(=O)Cc2c[nH]nc2O)CC1 N1(C(CC(CC)O)=O)CCC2(CCN(C(=O)C=Cc3ccncn3)CC2)C1 C1(CNC(C(C)(C)SC)=O)N(C(=O)C(F)n2ccnc2)CCC1(C)C c1(C(=O)NC(C)CNC(c2cn(C(F)F)cn2)=O)ccccc1N1CCOCC1 c1(SCC)cc(Cl)ccc1C(=O)NC(CO)C(C)NC(C1CCCN1C(C)C)=O CN(OC1CCCC1)C(=O)C(CC1CC1)NC(C1CC2(C1)CC2(F)F)=O C1(C(=O)NCC2(F)CCC(NC(CCCC)=O)C2)COc2cc(F)ccc2O1 C1(NC(CCC2(NC(CC3CCCN(C)C3)=O)CCC2)=O)CCCCNC1=O N1(C(C2C(C)CC=CC2)=O)C2CCC1CC(CNC(C1CC13CCOCC3)=O)C2 CC1=C(C(=O)NC2CCCN(C(C3CCCNC3=O)=O)C2)CCS1(=O)=O c1(C(=O)NC2CC(NC(CC(CC)C(F)F)=O)C2)cc(=O)oc2ccc(O)cc12 c1(C(=O)NC(C2N(C(C(CC)O)=O)CCC2)C)ccc(Cn2cccn2)cc1 CCC(C)C(C(=O)N1CCC2(CC1)CC2)N(C)C(C1C(C)C1C)=O N1(C(C(CC(=C)C)NC(C)=O)=O)CCCN(C(c2sc(OC)nc2Cl)=O)CC1C N1(C(c2c(C)nccc2)=O)CC2CC(C(N3CC(F)CC3C#N)=O)C(C2)C1 CC(C)CC(F)C(=O)NC1(C2CCCCN2C(=O)CCC(=O)N(C)C)CC1 c1(N2C(C)CN(C(C3(F)CCC3)=O)CC2)ncnn2cccc12 c1(OCC(=C)C)ccc(CCC(=O)OCCN2CCCC2CC(=O)O)cc1 c1(C(=O)NC2(C(=O)NCCCCCC3CC3)CC(F)(F)C2)cnn2ccccc12 Cc1cc2c[nH]nc2cc1C(=O)N(C)CCOCCN(C)C(C1CC(F)C1)=O C(=O)(C1=CCC(C)(C)CC1)NC(C1CCCN(C(=O)CSCc2cscn2)C1)C CC1CC(=O)CCC1C(=O)N(C(CC(N)=O)C(=O)O)Cc1ccccc1 c1(NC(C2CC2C(=O)NC(c2ccccc2)CO)=O)cnc(Br)cn1 c1(CNC(c2cccc(Cl)c2Br)c2n(C)nnn2)ccc2occc2c1 N1(N(C)C)CCCN(C(=O)NCc2ccc(Cl)cc2Cl)CC1 Cc1cc(C)c(CN2CCCC(NC(C34CCC(CC3)CC4)=O)CC2)c(C)c1 C(=O)(CN1C(=O)CCCc2sccc21)N(CC(CC)NC(c1ncn(C)n1)=O)C N1(C(C(=O)NCC)=O)CCCN(C(c2ccc(F)cc2C#N)=O)C(C)C1 N1(C(c2nc(CC)oc2C)=O)CC2CCC2(CCNC(=O)CCC#N)C1 C1(C(=O)NCCN(C(Cn2cc(CC(=O)OC)nn2)=O)C)CN2CCC1(C)CC2 C1(OC)CC(CNC(C2CC(O)C2)=O)N(C(=O)CC(F)F)C1 c1(C(N2C(CNC(c3cnc(C)[nH]3)=O)CC(C)(C)C2)=O)ccc(S(C)=O)cc1 N1(C(=O)OC(C)(C)C)CCC2(CCC2C(=O)NCC(=O)NC2CCC2)CC1 c1(NC(C)=O)ccccc1C(F)(F)C(=O)NC1CN(C(=O)C(C)=C(C)C)C1 c1(C(N(CCNC(C2CCC(C)NC2=O)=O)C)=O)ncn2cc(Br)sc12 c1(CC(N2CCC(NC(c3c(C)cco3)=O)(CF)C2)=O)coc2cc(O)ccc12 c1(OC)cc(Cl)ccc1C(=O)NC(C)(CNC(c1ccns1)=O)CC(C)C Cc1[nH]c2c(C(=O)NCC3OCCC3C(=O)O)cccc2c1C c1(CC(=O)NCC(CNC(C(C)C2CCC2)=O)F)ccc(OCC#N)cc1 C(C1=CCCOC1)N(C(=O)C(Cc1ccco1)NC(=O)CCC1(C)CC1)C CC1C(=O)N(C(c2nc(Br)cn2C)=O)CCN1CC1CCOC1 C1(C(=O)NC2COCCC2O)CC2CCN(Cc3c(I)ccnc3O)CC12 C1(c2cn(Cc3ccc(CNC(C4C(C)CC4)=O)cc3)nn2)CCC(C)(C)CC1 C(=O)(C1SCCc2ccccc21)NCCN(C(=O)CC1COCCO1)CC1CC1 C1(NC(C2C(COC)C2)=O)C2CC3CN(C(=O)CCSc4cccs4)C1C3C2 C12C(CC1O)NC(=O)ONC2=O.C1(C)(SC)CCCC1 C1(OCC)CC(NC(=O)C(CNC(c2nnc(O)nc2O)=O)OC)C12CCC2 c1(CNC(C(c2ccnn2COC)N(C(CC)CC)CC)=O)nnn(C)n1 Cc1cccc2c1ccn2CC(=O)NC1C=CCN(C(=O)C=CC(F)(F)F)C1 C1(C)(CC(=O)N(CC(CC)NC(=O)C(c2ccccc2F)C)CC)CC(F)(F)C1 C1(F)(CNC(C=C(C)C(C)C)=O)CCN(C(c2c[nH]ccc2=O)=O)C1 N1(C(c2c(NC(=O)OC)cccc2)=O)CCC(F)(F)C(CNC(=O)CC(F)F)C1 N1(C(c2c(C)nc[nH]2)=O)CCN(C2CN(C(=O)C(C)c3cccs3)C2)CC1 N1(C(C2=C(C)CC2)=O)CC(NC(=O)CC2(O)CCCN(C)C2)C(S(C)(=O)=O)C1 N1(C(CCCC=C)=O)CCN(C(C2CC(F)CN2C)=O)CC1CC N(C1CC2(CN(C(=O)C(C)(CC)C(N)=O)C2)n2ccnc21)C(CCCOCC)=O C1(NC(C=CC=CC)=O)CC(F)(CN(CC)CC)C1.C1(=O)C(CC)N1 Cc1cnc2ccccc2c1C(=O)NCCC(C)NC(=O)C(C)CF S(=O)(=O)(c1cccc(=NCC(C)Oc2ccc(F)cc2)[nH]1)NCCC(=O)NCC C1(C(C(=O)NC)N(c2c(F)ccc(OC)c2)C)CC2(C1)C(F)(F)C21CCC1 c1(C(=O)NCCN(C(c2c[nH]c(=N)s2)=O)CC)sccc1C(C)(C)C CC1=NNC(=O)C1CC(=O)NCC1(C(N)=O)CN(C(c2cc(C(=O)O)ccn2)=O)C1 Cc1ccn2ncc(C(=O)NC(C)CC3CN(C(C4(C)CCCC4C)=O)C3)c2c1 C1(C(C)C)C(=O)NCc2cn1nn2.c1(CC)nn[nH]n1.C(C1CC1)(C1CC1)SC N1(C(C)C)CCCN(Cc2ccnc(-c3ccc(-c4nn[nH]n4)cc3)c2)CC1 CC(C)S(=O)(=O)C1CCN(C(=O)CCn2cc(-c3ncnn3C)nn2)C1.C1CCC1 N1(C(C(CC)c2ccccc2)=O)CCC(C)(C)C1CNC(c1c(O)noc1C)=O N1(CC(=O)NCCC(CNC(CC2C(C)C2)=O)(C)C)C(=O)c2ccccc2C1=O C1(N(C)C)(C(N2CCCC2Cn2cc(CN3CCOCC3)nn2)=O)CCCSC1 N1(C(C(C)(C)OC)=O)CCC(CNC(=O)C(c2ccccc2Cl)(C)C)C(C)C1 c1(C(N2CC3(C(NC(C(CCC)OCC)=O)CC3)C2)=O)nc(O)nc(O)c1F C#CCCC(C(=O)OC)NC(=O)CCCCCBr C1(C2CN(C(=O)CCC3CC(C(=O)OC)CO3)C2)(NC(c2cn(CC)nn2)=O)CC1 CC1=NOC(CC(=O)NC(CNC(=O)CCc2ccc(C)s2)CO)C1 c1(CCC(=O)N(C2CCN(C(=O)OC(C)(C)C)CC2C)CC)ccc(F)cc1Cl N1(C(C2CCC(C)(C)CO2)=O)CC2(CCN(C(C3(C(C)(F)F)CC3)=O)C2)C1 CC1CN(C(C23CCCC(C2)OC3)=O)CC2(CCN(C(=O)CCC(N)=O)CC2)O1 CC(C)(C(=O)N1CC(c2nc(-c3cc(OC(F)F)cc(F)c3)no2)C1)S(C)(=O)=O C1(NC(=O)NCCOC2COC2)CCCN(C2CCCC2)C1 c1(N(CCC#C)CCCOC)ccc(OCc2ccccc2)cc1 c1(C(N2CCC(O)(CNC(C(C)CF)=O)C2)=O)ccc(=O)n(CC(F)(F)F)c1 C12(NC(C(CCCC)O)=O)CCC(CC1)N(C(c1cnnn1C1CC1)=O)C2 C(=O)(CCCC(C)(C)C)NCC1CN(C(C2(CC)CC=CC2)=O)CC1C(F)(F)F C#CCCC(C(=O)NC(C(=O)OC)C1CCC1)NC(C1C2CC3C(C2)C13)=O CN1CCN(C(C2CC2CNC(=O)C=CC(N)=O)=O)CC1CC1CC1 N1(C(c2cnc(C3CC3)s2)C(=O)NCCC2CC2)CCS(=O)C2(CCC2)C1 O=S(=O)(c1ccc(NCC2(F)CCOCC2)c(F)c1)NC1CCOC12CCCC2 CC1CCNCCC1N(C(C1(C(F)(F)F)CC1)=O)CC1CCCCO1 C(=O)(C(C)(C)C(F)F)N(C1CCCN(C(c2nn(C)cc2Cl)=O)C1)C C1(N(C(=O)C(C)CSc2ccc(F)cc2)CC)CCN(CCC(=O)NC)CC1 C1(C(N2CCCC(CNC(C(F)=CC)=O)C2)=O)COc2c(OCC)cccc2C1 c1(C(=O)NC(C(C)C)CNC(C2CCCCN2C(C)C)=O)ncnc2ccsc12 C1(F)(C(=O)OC)CC(C(=O)NCCCNC(=O)CC2CCCCC2)C1 C1(CC(=O)Nc2cccc(NC(C(C)OCC)=O)c2)CCC2(CCC2)CO1 N1(c2nc(N(CCCSC)C)nc(C)c2)CCn2c(nn(C)c2=O)C1 c1(C(=O)NCCCCCNC(C2(C#N)CC3CC3C2)=O)nccc2ncncc12 c1(C(N2CC3C(NC(Cc4c(C)ncs4)=O)(C3)C2)=O)cnc2ccsc2c1 c1(C(=O)NC2CCCN(C(C(CC)C(C)(F)F)=O)CC2)oc2ccccc2c1C C1(C#N)(C(=O)NCC(CC)NC(=O)C(C)C(C)C)CC2(CC2)C1 C=CCCCC(C(=O)NC1(C)CC1(C)C)NC(=O)Cc1c(C)noc1C c1(CC)nc(C(=O)N(CC(C)O)CC2CC2)c(C)o1.c12ccoc1C(=O)NC2 N1(C(C2C(C)N(C)CC2)=O)CC(C(N2CCN(C)CC2CO)=O)C(F)(F)C1 c1(C(=O)NCC#CCNC(C2CCC(C)(CC)O2)=O)cc2ccccc2nc1O CCCCCCCC(=O)NCC1COCC1NC(c1ccc(Br)o1)=O c1(C(N2CCC(C(C(=O)N(C3CCOC3)CC)C)C2)=O)ccncc1NC CCCCC(C)CCC(=O)N1CCC(NC(c2cccc(N(C)C)c2)=O)CC1C C1(C(=O)NC2C(NC(C3CSC3)=O)COCC2)Cc2nnsc2S1 C(CNC(=O)CCN1CCOC1=O)(CC(=O)Nc1cc(C(N)=O)nn1C)OC CN1CC(O)CC1C(=O)NCc1csc(C(=O)N(CCO)CCO)c1 c1(C(CC)Cc2ccc(C(F)(F)F)cc2)nc(-c2ccc(C)o2)nn1CCOC C12(CN(C)C)CC(CN1C(C1CC(NC(=O)CCCN(C)C)C1)=O)C2 c1(CNC(CCC2CC(C)C2)=O)ccoc1C(N1CC=CCC1)=O C1(C(N(CCCCNC(=O)Cc2csc(Cl)n2)C)=O)CCCC(F)C1 C1(CCOC)CN(C(c2ncoc2C2CCC2)=O)CCN1C(=O)CP(C)(C)=O c1(C(=O)NC2COCCN(C(=O)C=Cc3ccoc3)C2)cn2ccc(Cl)cc2n1 CCCCC(CNC(c1cncc(COC)c1)=O)NC(c1cc(C)n(C)n1)=O C(=O)(C1Cc2ccccc21)N1CCC(CC(=O)Nc2ccc3cc[nH]c3n2)CC1 c1(SC)cc(C(N2CCC(O)(CNC(c3ccc(F)o3)=O)C2)=O)ccc1F O(NC(=O)C(O)CNC(=O)CC1CCCC1O)CC(CC)C Cc1cc(Br)ncc1NC(C1CCN(C(c2ccc(F)cc2)C)C1=O)=O Cc1cnc(NC(c2cscn2)CO)c(S(=O)(=O)NC(C)CO)c1 N#CC1(C(=O)NC2CCC(NC(C3(C(F)F)CCCO3)=O)CC2)CCOC1 C(C)(CNC(C1(C)CC1(C)C)=O)(CC(C)C)NC(CCc1ccc(C)cc1)=O c1(C(=O)NCC(CNC(c2ncc(Br)cn2)=O)OC)cnc(O)n1C C(C(C)(C)CC(=O)NCCC1CC(NC(c2ccc(Cl)nc2OC)=O)C1)OC Cc1ccc(C(C)C(=O)NC2CC(NC(c3ncncc3Br)=O)C2)cc1 N1(C(CSc2ccc(C)cc2)=O)CCCN(C(C2CSC2)=O)CC1C C12(C(N(CCCNC(C(n3ccc(Br)n3)C)=O)C)=O)CC(F)C1C2 c1(-n2cc(C3(C)CCCC3)nn2)cccc(C(=O)NCCc2cccnc2F)c1 C(CC(C(=O)N1CCC(C#N)C1)NC(=O)CCCOC)OCC C12CCC3(CC1)CC(C3)CN2.C1(C(=O)OC)CN(C(=O)OC(C)(C)C)C2CC12 S(=O)(=O)(c1c[nH]ccc1=NCc1ccc(Cl)s1)NC(C)C(C)CO CCC(CN(C)C)CC(=O)NC(C1CCN(C(c2ccc(C(C)=O)[nH]2)=O)C1)(C)C c1(OC)ccc(CCCC(=O)NC2COCC2NC(=O)C(C)C(C)O)cc1 N1(C(=O)Cc2ncc(Cl)s2)CC2(C1)CN(C(c1cn3ccccc3n1)=O)CCO2 C1(CNC(c2cc(CCCO)on2)=O)CN(C(=O)C(F)F)CC1C(F)(F)F N1(C(C(CC=C)C)=O)CC2CCC1CC2NC(=O)C(F)(F)C1(O)CCC1 c1(C(=O)NCC(=O)OCC(=O)N(CCC(=O)NCC)C)cn(C)cc1C C(CCCCC(=O)NC(c1cn(C)nn1)C(=O)NCc1ccc(F)c(F)c1)OC N1(CC(=O)NC(CCCCCC)C)Cc2c(C(=O)O)ccc(F)c2C1 N1(C(CCN(C)CC)=O)CCC2(CC1)CCN(C(=O)CC1CCC(C)O1)C2 c1(C(=O)OC)c(C(=O)NCC(C2CCOC2)NC(C2CCCCC2)=O)n[nH]c1C C(=O)(C1=C(F)CN(C(C2C3CCC(C3)C2C)=O)CC1)NCCCCCC C1(CNC(C2(C)CCC2)=O)CC2CC(C1)N(C(c1cnn(CC(F)(F)F)n1)=O)C2 C1(CC)(NC(=O)Cc2cccc(C(F)(F)F)c2)CCN(C(=O)C)CC1.OC C1(=O)C(C)(C)CN1.c1(C(=O)OC)ccccc1Cn1cc(CC(C)O)nn1 C(=O)(CCCCC(C)C)NC(C(C)NC(c1n(CC)cc(Br)c1)=O)C C(=O)(C(CCCOC)NC(c1c[nH]c(C(N)=O)c1)=O)NCC=C c1(N2C(CCNC(C(CCC)CCC)=O)CSCC2)nc(C)c(C#N)cc1Cl c1(CCCC(C)SC)nc(CCN(C)C)nn1-c1cnn(C)c1 c1(C(N2CCC(C)(CC(=O)NCC(c3ccco3)O)C2)=O)cc2occc2[nH]1 O=C1NC(Cc2ccc(F)c(Cl)c2)C(=O)N1Cc1cccc(-n2cncn2)c1 C(=O)(C(C)(CO)NC(c1nc(CC)oc1C)=O)N1CC(C)(CC=C)C1 CCC(C(=O)N(CCN(C)C(c1cnn(C2CC2)c1)=O)C(C)C)OC1CCCC1 N1(C(=O)NC(C(=O)OCC=C)C(C)C)CCC(O)C(CN(C)C(C)C)C1 c1(C(=O)NCCCNC(=O)CNC(c2ccncc2)=O)ccc(C2CC2)cn1 c1(OC)nc(C(=O)N(C(C)CCNC(C2COC(=O)O2)=O)C)sc1C c1(OC)ccc2c(Nc3cc(-c4ccc(OCC)cc4F)ccn3)ncnc2c1 Cc1ccn2cc(C(=O)N(C(C)CNC(=O)C=C3SCC(=O)N3C)C)nc2c1 c1(C(=O)NC2CN(C(CCC=C)=O)C(C)C2)c(Br)c(C)nn1C C1(C(=O)NC(C)CCC(F)F)CC2(CCCCC2)C1 N1(C(c2ccc(CCCCC)cc2)=O)CCC(NC(=O)C(C)C2CC2)CC1C CC(C)CCCC(=O)NCCC1CN(C(=O)CCCn2ccnn2)CC(C)O1 C1(C2CN(C(=O)CCCCn3ccnn3)C2)(NC(c2csc(O)n2)=O)CC1 C(=O)(C(C(C)(C)C)n1ccnn1)N(CC(CNC(CN1CCC(C)CC1)=O)C)C c1(OC)ncc(Cl)cc1C(N1CCCC(N(C(=O)C(C(C)C)OC)CCO)C1)=O C=C(C)CC(C)C(=O)N(C1CN(C(c2oc(C)nc2CC)=O)C1)C c1(C(N2CC(C#N)N(C(c3ccncc3)=O)CC2)=O)ccc([N+](=O)[O-])c(F)c1 C1(NC(C(C2CC2)OCC)=O)CCCC1CNC(=O)Cn1cnnc1C1CCC1 C1(C(=O)NC2(CC=C)CCC2)CC2CN(C(=O)C(C)(C)C(=C)C)CC2C1 N1(C(c2c3ccc(C)cc3sc2)=O)CCC(C2CCN(C(C3COC3)=O)CC2)C1 C1(C(=O)NC2C(NC(Cc3c(C)non3)=O)CCC2)Cc2ccccc2S1(=O)=O c1(C(N2CCC(NC(CC3(C)CCC3)=O)C2)=O)cccc2ncsc12 N1(C(C(C)SC)=O)CCC(C)C(N(C(=O)CCCCCNC(C)=O)C)C1 c1(N(CC(F)F)C)nc(=NCCc2ccsc2Cl)[nH]c2c(F)cccc12 c1(C(=O)OC)cccc2c1CCC2NC(=O)N(C)Cc1c(I)cnn1C c1(C(=O)NCC2C(NC(CSc3n(C)ccn3)=O)CCC2)c(N)cc(F)cc1Cl C1(NC(Cn2nc(C)oc2=O)=O)CN(C(c2ncccn2)=O)CC1C1CC1 c1(OC)cncc(CC(=O)NCC2CCC(NC(C3CCS(=O)CC3)=O)CC2)c1 CC1(NC(c2cc(O)nc(C3CC3)n2)=O)CCN(C(C2CCCCO2)=O)CC1 c1(C(N2CC3C(NC(=O)CC4CC5CC5C4)(C3)C2)=O)cnc2ccccn12 c1(C(=O)NCCCOCCNC(C2(CC#C)CCCC2)=O)ccc(P(C)(C)=O)o1 C(=O)(CCC(C(=O)O)NC(c1ccc(F)cc1C(F)(F)F)=O)N(C)C C(=O)(C(=O)C(C)(C)CC)N1C(CCC)CN(C(=O)Cn2cc(C)ccc2=O)CC1 c1(C(=O)NC2(C)CN(C(Cn3ncc(C)c3)=O)C2)cn(C)c2ccccc12 C12(CNC(C(C)(c3cccs3)OC)=O)CCC(CC1)N2C(C1CN(C(N)=O)C1)=O C1(CNC(C2C3COCC23)=O)(CO)CCCN(C(C2C=CCS2)=O)C1 c1(OC)cc(N(C)Cc2cnc(N(C)C)nc2)ccc1NC(C)=O C1(C(=O)NC(CCN(C)C(c2n[nH]c(=N)[nH]2)=O)c2cccs2)COC(=O)C1 c1(SCC)ccc(C(=O)NC2CCN(C(=O)C(C)COC)C2C2CC2)cc1Cl Cc1cccc2c(C(N3CC(O)CC3c3cc(F)ccc3F)=O)nccc12 C1(C(=O)NC2CCN(C(c3ncc(CC)s3)=O)C(C)C2)CCCC1S(C)(=O)=O C(=O)(C(C(C)O)N(C)C)NCC1(OC)CN(C(c2cc(C3CCCC3)[nH]n2)=O)C1 N1(C(CNC(CC(C)(C)C)=O)=O)CC(NC(c2cnn[nH]2)=O)Cc2ccccc21 N1(C(C(C)O)=O)CCc2ccc(-c3cc(F)c(O)c(F)c3)cc2C1 N1(C(C2CCN(C(C)C)CC2)=O)CCC2C(CCCN2C(c2cccs2)=O)C1 c1(C(=O)NC(C2CCOC2)CNC(=O)COC2CC2)cc2ccccc2o1 N1(c2nccc(OCCOC)n2)CC(NC(c2ccnc(C)n2)=O)C(C)(C)C1 C1(OC)CC2(C1)CC(C(N1CCN(C(=O)CCc3ncccn3)C(CO)C1)=O)C2 C1(CNC(=O)NCC(Cc2cccnc2)CO)CCCCC2(C1)OCCO2 C1(C(=O)NC(C(=O)OCC)CO)CSCCN1C(=O)CN1CCCC1 c1(SC)ccccc1C(=O)NC1CCOCC1NC(=O)CCCn1ccnc1 CC1CCC(CC(=O)NCC(=O)NC2CCC(SCCO)CC2)OC1 CCC(C)C(O)C(=O)NCCCC(C)NC(c1c(OC)nsc1OC)=O c1(C(N2C(CNC(=O)C=Cc3ccccc3)CCCC2)=O)n[nH]c2c1CC1CC21 Cc1nc(C(C)(C)C)ncc1C(N1CCCCC1CNC(c1cnoc1C)=O)=O C(C(=O)NCC1(C(N)=O)CN(C(=O)C(c2ccccc2)C)C1)(C(C)C)SCC N1(C(CC(C)(F)F)=O)CCC(C2CCN(C(c3cc(C4(C)COC4)no3)=O)C2)C1 N1(C(CS(CC)=O)=O)CC(CNC(c2ccc(OC3CCC3)cc2)=O)C(C)(C)C1 CC1=NN(C)C(=O)C1CC(=O)NCCOCCNC(=O)CC1CCOC1C N1(C(c2c(OC)nsc2)=O)CCC(NC(=O)C(=Cc2c[nH]cn2)F)C(F)(F)CC1 N1(C(c2c(Br)c(C)n(C)n2)=O)CC(CNC(=O)CC(C)F)CC(C)(C)C1 C1(C(=O)NCC(CNC(CNC(C)=O)=O)C(F)(F)F)CCn2ncnc2C1 CS(C)(=O)=NC(=O)C(=O)NCC1CN(C(c2c[nH]nc2C2CCOC2)=O)CC1O c1(OC)cc(C(N2CC(F)CC2CN(C(=O)C(F)OC(F)(F)F)C)=O)ccc1Cl c1(OC)ccccc1C=CC(=O)NC1CCC(NC(=O)C(F)CC2CCC2)C1 N1(C(c2ccc(C(C)(C)C)s2)=O)CC(NC(C2CCCO2)=O)CC(O)C1 c1(C(C)NC(=O)CCNC(=O)C(=O)N(C)C)ccccc1NC1CC(=O)N(O)C1 Cc1ccc(F)cc1CC(=O)NC1CN(C(=O)C(O)c2ccsc2)CC1C N1(C(CC(=O)NC)=O)CCC(C)N(C(C2CC=CCO2)=O)CC1 c1(SCC)ccc(C(=O)NCCOCCN(C)C(C2CNC(=O)N2)=O)cc1 c1(C(=O)NC2CCC(NC(Cc3cccc(CC)c3)=O)CC2)ccc(C)cc1C N1(C(C(C(=O)OCC)F)=O)CCCC(CCNC(=O)C(C(C)CC)N(C)C)CC1 c12ccc(cc1)NC(C(C)C)CNC2=O.c1(C(C)=O)cccc(NC=O)c1 C1(C(=O)NC2(COC)CN(C(C3CCCN(C(C)=O)C3)=O)C2)CCCC(F)(F)C1 c1(C(N2CC(CCO)C2)=O)cc(Cl)cc(S(=O)(=O)N2CCOCC2)c1F C(=O)(C1=Cc2ccccc2OC1)N1CC2N(C(c3csc(C)c3C)=O)C(CC2)C1 C(=O)(CC(C)(C)C)N(CC(C)NC(=O)C=CCCc1ccccc1)CCOC CC1(C)COC(C(=O)NC(CNC(c2ccccc2OCCF)=O)C2CCC2)C1 C(=O)(C1=NOC2(CNC2)C1)N1C(CC)CN(C)C(=O)C1 CCCCC(CCCC)(c1nnnn1CCSC)NCC1CCC2(CC2)C1 C1(NC(c2ccc(C)s2)=O)C2CC3CN(C(C4CC(C)OC(C)C4)=O)C1C3C2 C(=O)(C(F)(F)C(O)C1CC1)NCC1N(C(c2ccc(C(C)C)cc2)=O)CC(F)C1 C1CC2C=CC1C2.C(CC(=O)OC)N(C(=O)CONC(=O)C1CC1COC)CCC CC(C)(C)CCC(=O)NC1C2CCN(C(C3CCS(=O)(=O)C3)=O)CC12 Cc1cn2c(n1)CCC(C(=O)NCC1CN(C(=O)CCOC3CC3)CC13CC3)C2 c1(NC(CCC23N(C(=O)OC(C)(C)C)CCC2C3)=O)ccc(F)c(Cl)c1F C(C(=O)Nc1ccccc1)(C(C)(C)C)NC(C=Cc1c(C)n[nH]c1)=O C1(NC(C(=O)NCC)=O)CCN(C(C)(C)C)CC1OC(C1CSC(C(C)C)C1)=O C#CCC(C)(C(=O)NC1CCN(C)C1)NC(C1CCCC1)=O C1(CC(=O)NC(C2CCOC2)C#C)C(NC(c2ocnc2C2CC2)=O)CC1O CC1(C)CC(CC(=O)N(C2CCCC2)CCCc2ccn(C3CC3)n2)C(=O)O1 C1(C(=O)NCC2N(C(C=CSC)=O)CC(C)(C)C2)CCc2nnn(C)c2C1 c1(C(=O)NC2CCCCN(C(C3(C)CCCO3)=O)C2)cccn2nncc12 C(=O)(C(=O)N=c1cc(C)o[nH]1)NC1CN(C(CC(C)OC)=O)C2C1CCC2 c1(C(=O)NC2(CNC(C3CC4(CSC4)C3)=O)CCC2)[nH]c2ccccc2c1Cl c1(C(=O)NCC2CC3CC3N2C(C2CC(F)(F)C2)=O)cc2cccn2cn1 C1(C)(NC(c2c(OC)cccn2)=O)CCN(C(c2cn(C)c(O)n2)=O)CC1 CCCCCC(C(=O)NC1CC2CN(C(=O)C(C)(C)c3nccs3)CC12)C(C)C c1(OC)cc2[nH]c(=N)sc2cc1C(=O)NC1CCC2CCC12 C1(NC(C(C2CCN(C(c3cc(C)sn3)=O)C2)C)=O)C2CCC(C2)C1CO Cc1cncc(S(=O)(=O)NC(c2cc3cnccc3o2)C)c1 c1(C(N2CCOCC(NC(C(C(C)C)C3CCC3)=O)C2)=O)ccc2c(c1)CCO2 N1(C(C=C(CCC)C)=O)CCCC(C(C)(C)C(=O)NCC(O)C(F)F)C1 C#Cc1ccc(C(=O)NCC2(OC)CCN(C(c3c(Cl)noc3C)=O)C2)nc1 C(=O)(CC(C)CCC(=O)Nc1cnn(Cc2ccccc2)c1)OC c1(OC)ccc(N)c(C(=O)NC23CC2CN(C(c2nncn2C2CC2)=O)C3)c1 Cc1cnc(C(=O)NCCOC2CN(C(C3(C)CCCCC3C)=O)C2)cc1C#N c1(OC)ncc(C(=O)NOCC23CCC(C(=O)O)(CC2)C3)cc1Cl C(CN=c1[nH]c(=N)[nH]c(=NC2CC3CCCCCC23)[nH]1)c1scc(C)n1 N1(C(c2cc(SC)c(N)cc2)=O)CCC2(CC(NC(=O)C(C)(F)C(C)(C)F)C2)C1 Cc1ccc2[nH]c(C(=O)NCC3(F)CN(C(c4ccc(Cl)s4)=O)C3)cc2c1F N1(C(C(C(=O)OC)C)=O)CC2CCC2(CC(=O)NCC2(C#N)CCOCC2)C1 C1(F)(CNC(CC2(C=C)CC2)=O)CCC(NC(c2cncn2C)=O)C1 O=C(C1=Cc2c(ccc3ccccc23)OC1)OCC1CCC2(CC1)COCCO2 N1(C(C2(NC(C(C)NC(CC)=O)=O)CCC(C)(C)C2)=O)CCC(=O)N(C)CC1 C(C(C)(C)CCCC(=O)OC)NC(C(=O)NCCC(CC)C)=O FC1(F)CC(n2nnnc2C2CC(NCC3CC(c4ccccc4)C3)C2)C1 C1(NC(C2C(C)CCC2)=O)CCN(C(=O)Cn2ccccc2=O)C1(C)C c1(CC(=O)NCCC2CCCN2C(=O)C(O)C(F)F)ccc(F)cc1 N1(C(CC2ON=C(C)C2)=O)CC=C(CNC(C2CC2(F)F)=O)CC1 Cc1cc(Cl)c(O)c(NC(c2ccc3nnn(C)c3c2)=O)c1F N1(C(C2(C#N)CC2)=O)CCc2cc(C(=O)Nc3ccnc4ncnn34)cnc2C1 c1(C(N(CC(CNC(C(CC=CC)CC)=O)O)C)=O)cnc2ccnn2c1C CC1CCCC1(C)C(=O)NC1C2CC(NC(c3ccc(Cl)cc3)=O)CC12 c1(NC(c2n(C(C)(C)C)nnn2)C2CCCSC2)cnc(Br)c(C#N)c1 C(CCCC(CO)NC(=O)C(c1ccccc1)N(C)C)NC(c1scc(C)c1)=O Cc1noc(C)c1CC(C)C(=O)NC1CCC(F)(CNC(=O)Cc2ccoc2)C1 c1(C(N(CCCNC(C2CC23CC3(F)F)=O)CC)=O)nccc2ccsc12 c1(C2C(C(N(CC(CNC(COCC(=C)C)=O)C)C)=O)C2)ccncc1 C(=O)(CS(C)(=O)=O)NCC(=C)CCNC(=O)CCSCc1ccccc1 C(C(CC1CCCC1)C(=O)NCC(Cl)Cl)NC(C(C)OCCOC)=O C(CCCCC(=O)N1CCC(NC(=O)C2=COCCO2)CC1)NC(N)=O N1(C(CCS(N)(=O)=O)=O)CCN(C(=O)C(F)CC2CC2)CC(O)C1 C1(C(CNC(C(C)OCCC=C)=O)(C)NC(C2CC(F)C2)=O)CCCCC1 C1(NC(COC(C)C)=O)CC2CC1CN(C(=O)CCc1cccc(C(N)=O)c1)C2 C(=O)(CCCC(F)(F)CO)NCC1CCC(NC(C(C)(O)c2ccccc2)=O)CC1 c1(C(N2CC(NC(CN(C)C(N)=O)=O)C(C)(C)CC2)=O)cc(F)cc2nn[nH]c12 C(CC(C(=O)N(C)Cc1ccc(F)cc1)NC(C1CCCC1OC)=O)OCC c1(N(C)C)cc(C(=O)NC2(CO)CN(C(C3COC(C)(C)C3)=O)C2)cc(Cl)n1 C1(CNC(c2n[nH]c(C)c2C)=O)CC(C)CN(C(=O)C=CC2CCOC2)C1 CS(=O)(=O)CCCC(=O)NCC1COCC1NC(c1cccc(C(F)(F)F)c1)=O N1(C(Cc2c(C)nn(C)c2)=O)CC(NC(=O)C(C)CC(C)(C)C)C(S(C)(=O)=O)C1 C(=O)(C1CCCn2nccc21)NC1CCCN(C(CCCCCOCC)=O)CC1 CCC(CNC(=O)CCc1nc(=N)[nH][nH]1)(CC)C(=O)NCC1CCC(O)C1 C(=O)(C(=O)C(C)(C)C)NC(CCNC(CSC(C)C)=O)(C)C C1(CC)CCCN(C(=O)NC)C1C(=O)NOC(c1ccc(Cl)cn1)C Cn1nc(C(=O)OCC2CCC(NC(=O)C3CC3)C2)c2ccccc12 C(=O)(C(F)(F)C(O)CC)NCCCCCN(C(c1nc(CC)sc1)=O)C(C)C CC1(C)CC2(CC(C(=O)NCCC3=CCN(C(=O)C(C)CC(N)=O)CC3)C2)C1 c1(OC)ccc(F)c(NC(C2(C)CN(C(c3cccc(Br)c3)=O)C2)=O)n1 N1(C(c2cn(CC)nc2)=O)CCOCC(CNC(c2c(C)coc2C2CC2)=O)C1 C(=O)(CC(C)CC(C)C)NCCCN(C(c1c(CC)cccc1F)=O)C N1(C(c2ncn(CC)c2)=O)CC=C(CNC(c2nnc(O)cc2O)=O)CC1 C(=O)(C(F)(F)C(F)(F)F)Nc1cccc(NC(C2CCN(OC)CC2)=O)c1 N1(C(COCC=C)=O)CC2(C1)CN(C(c1ccc(-c3ccncc3)o1)=O)C2 N1(C(c2c(C)nc(CC)s2)=O)CCC(C)(C)C1CNC(C1(O)CCCCCC1)=O C1(NC(c2ccc(C#C)o2)=O)CC2CCC(C1)N2C(=O)CC(C)CC(C)C C(=O)(C1=CC2CCC(C1)C2)NC(C(=O)NCC(C)CN(C)C)C1CCC1 CCC(C)C(C(=O)N(CCCNC(c1cnncc1O)=O)C(C)C)NC(=O)OC c1(OC(C)C)ccc(C(C(=O)OC(C)(C)C)N(C)CCn2ccnc2)cc1F N1(C(C2(C#C)CN(C(=O)CCCCC)C2)=O)CC2(CCC2)C12CCC2 C(C(O)CC(F)(F)F)NC(C1C2(CC(NC(CCCOCCC)=O)C2)C1)=O c1(C(N2CCC(NC(c3cnc(O)c(F)c3)=O)C2)=O)cccc(S(=O)(=O)CF)c1 c1(C(N2C(C)CN(C(C3CCSCC3)=O)CCC2)=O)cc2c(nn1)CCCC2 c1(C(=O)NCC2OCCN(C(CC3CCCN(C)C3)=O)C2)cc2cccnn2n1 c1(C(C)NC(C(=O)N(C2CCC(C)C2)CCO)=O)ccc(Cl)cc1 c1(CC(=O)NC2(C)CC(NC(COCC(=O)OC)=O)C2)nc2c([nH]1)CCCC2 c1(C(N2CCC(NC(c3nn(C)c(O)c3)=O)C(F)C2)=O)ccc(I)c([N+](=O)[O-])c1 C1(C(=O)NC(C(=O)NCC2(CO)C(C=C)C2)c2ccco2)CC2(CC2)CO1 N1(C(C2(COC)CC=CC2)=O)CC(N(C)C(c2nncs2)=O)C2(CC2)C1 c1(C(C)NC(=O)CC(N)Cc2cccc(F)c2)cc(Cl)ccc1OC(F)F C1(C)(C(=O)NCC2C(NC(CCc3c(C)noc3C)=O)CC2)CCCNC1=O Cc1[nH]c2ccncc2c1C(=O)OC(C)C(N1CCN(c2ncccn2)CC1)=O Cc1cnc(C(=O)NC2CCC(CCNC(C3(F)CCCOC3)=O)C2)cn1 N#Cc1ccc(CN2CCC2C(=O)Nc2cccc(CCO)c2)cc1Cl CCC(CC)C(C)C(=O)N1CC2CCC1C(NC(C1CC3(CC3)C1)=O)C2 N1(C(CCOCC#C)=O)CC2=C(C1)CN(C(c1occc1COCC)=O)C2 c1(C2(C(=O)NCCCOCCNC(=O)CN3CCCC3=O)CC2)ccc(F)cn1 N1(C(c2n(CC)nc(C)c2)=O)CC2CC1CN2C(=O)CNc1c(C)cccc1C c1(N(CC(C)CNC(=O)CC2COCC(C)(C)O2)C)ccnc2ncnn12 c1(C(=O)NCCCN(C(C2C(C(=O)OCC)C2)=O)C)nc(C)c(C)[nH]c1=O c1(C(=O)NC2CCN(c3nccc(C)n3)CC2F)cccc2c1CC(=O)N2 C1(C)(CNC(CC2CCN(OC)CC2)=O)COCCN(C(=O)C(C)(CC)CO)C1 C(=O)(CC(C)C(=O)NCC(C)C(=O)NCc1ccnc(CO)c1)OCC N1(C(C2C(C=C)OCCC2)=O)C2CCC1CC(CNC(=O)COCCN(C)C)C2 C1(C)(C(=O)NC(CC)CC)CN(C(C2CCCN(C)C2)=O)C(C)(C)C1 C(N=c1[nH]c(=NC(C)c2ncnn2C)c2[nH]ccc2[nH]1)c1ccc(SC)nc1 Cc1noc(C)c1C(N1CCC(CCC(C)O)CC1)C(=O)Nc1ccccc1Cl c1(C(N(CCOCCN(C)C(c2cc(CO)[nH]n2)=O)C)=O)c(O)cc(Cl)cc1F Nc1ccccc1NC(=O)Cc1cccc(C(=O)NCCC(=O)OCCO)c1 C1(NC(c2n(CC=C)ccc2)=O)CCC(C)(CNC(c2cscc2SC)=O)C1 c1(C(=O)NC(C2N(C(C3CC(N(C)CC)C3)=O)CCC2)(C)C)cc(Cl)ccc1F C=CC(C)CC(=O)NC(CN(C(=O)C(C)NC(=O)CC)C)CC O=C1CCCC(C(=O)NC(CCC2CC2)C(=O)N2CC(F)C(F)C2)CC1 C1(C(=O)NC(CC(C)NC(=O)CN(C)C)C)CCN(c2nccs2)CC1 c1(C(=O)NCC(CNC(C=C(COC)C)=O)CO)cc(C)cc(OC)c1O N1(C(C(CC=C)OC)=O)CC2CN(C(C3(NC(C)=O)CCCC3)=O)CC2C1 Cc1ncccc1-n1nc(CCN(C)C)nc1-c1cnc(C(C)C)o1 C(=O)(C1=CCCOCC1)N(C(C)C)CCNC(C1CC(=O)C1C(C)(C)C)=O N1(C(C2(C)CCN(C)C2)=O)CC2CN(C(c3ccn(C4CC4)n3)=O)CC2(C)C1 N1(C(CC(=O)NCC)=O)CC(NC(C2(C)CC(C#N)C2)=O)CC12CCCC2 N1(C(CN(C2CC2)CC)=O)C(CNC(c2cncs2)=O)CC2CC12 N1(C(CONC(=O)CCC2CC2)=O)CCc2n[nH]cc2C1 CCCCC(CC)CC(=O)NC1(C)CCCC1NC(=O)CCC1CCCC1 c1(CC)cccc(C(N2CCOCC(CNC(c3ncncc3F)=O)C2)=O)c1N Cc1cc(C(=O)NCCC2(NC(=O)Cn3nccc3C(F)(F)F)CC2)co1 CCN=C(NCc1ccn(C)c1)NC1Cc2ccccc21 Cc1nc[nH]c(=NCC2CN(C(=O)Cc3nc(C(C)(C)C)cs3)C2)c1Br C1(F)(C(=O)NCC(=O)NCC(=O)NCc2ccn(CC)n2)CC=CCC1 C1(C(=O)NCCCCCN(C)CC)CCC2(CC2)N1C(=O)C(C)S(N)(=O)=O C1(NC(CCCOCC)=O)CCN(C(C2CCC(=O)N2)=O)C1C(C)C CCCC(C(=O)NCc1ncoc1C1CN(C(c2ccn(C)c2)=O)C1)OC C1(CC=C)(NC(=O)CCc2ccccc2)CCCN(C(=O)C(C)NS(C)(=O)=O)C1 c1(-c2nc(CC3(OC)CCC(=O)CC3)nn2C2CC2)cnc2c(c1)CCOC2 c1(C(=O)NC2CCC(NC(=O)CNc3cccnc3)CC2)cnn2ccncc12 CC(CSC(F)(F)F)C(=O)OCC1CCCN1Cc1cccnc1 C1(CNC(c2ccc(C)nc2)=O)CC2(CCN(C(c3nnccc3C)=O)C2)CO1 C1(NC(CCc2cc(C)no2)=O)CC(C(=O)NC2C3CCC2CC3)C12CCC2 C(=O)(C(O)C(F)(F)F)N(CC(CN(C(c1cccc(OCC)c1)=O)C)O)C c1(Nc2c(NC(=O)OCC)ccc(C)n2)ccc(N2CCCC2)c(C#N)c1 c1(-c2nc(-c3cc(OCC)ncc3)nn2-c2cccnc2)ccc(CC)nc1C c1(-c2scc(-c3nc(C4CC(O)CN4C4CC4)on3)n2)ccc(I)c(Cl)c1 c1(C(=O)NC(C(C)NC(C(CCOC)C)=O)(C)C)ccc2[nH]c(=N)n(C)c2c1 N1(C(C(F)=CCC)=O)CC(NC(C2CC(C)(C)CO2)=O)CC1(C)C N1(C(CC(=C)C)=O)CCC(O)(C2CCN(C(C3CN4CCN3C(C)C4)=O)CC2)C1 Cn1ncc2c1CCCC2N=c1[nH]c(=NCC2CC(F)C2)[nH]c2c1CCCCC2 N1(C(c2nc(C(C)(C)C)oc2)=O)CC2CN(C(c3ccccc3Cl)C)CC2C1 C1(C(=O)OC)CC1C1CN(C(=O)CC2OCCO2)C1.C1(=O)CO1 c1(C(N2CC(CNC(c3ccnc(OC)n3)=O)C2)=O)n[nH]c2c1CC1CC21 N1(C(C=Cc2nc(C)c(C)[nH]2)=O)CC2CCN(C(=O)CC3(O)CCC3)CC12 c1(C(=O)NC(CC=C)CNC(=O)C(C)c2ccsn2)cc(C)c(F)cn1 C1(CNC(C(C)C2CC2)=O)CN(C(=O)CC2CCC(F)(F)CC2)CCC1(F)F Cc1cc(N2CCn3nnc(N)c3C2)nc(=NCCOCCNC(C)C)[nH]1 C1(OC)CCCCC1n1nnnc1N1CCCC(c2n[nH]cc2C)C1.C(C)(C)C C(C(C)(C(=O)NC1CCC(C(=O)NCc2nccc(C)n2)CC1)OC)OC c1(C(N2CC(NC(c3c(CC)occ3C)=O)C3C2C3)=O)ccc(C)c(N)c1 C12(NC(c3cncc(C(C)(C)C)c3)=O)CCCC1CN(C(=O)CN1CCCC1)C2 C(C)(CCC(=O)NCCN(C)C(c1cc(OC)cnn1)=O)OC C1(CNC(C(CSC)O)=O)COC(C)(C)CN1C(c1ccc(OC(C)C)nc1)=O C1(NC(C2CC(C)(NC(=O)CCc3csnn3)C2)=O)CC2(CCC2)C1O O=C(C1=CCOC1)NCC(CNC(c1cscc1C1CC1)=O)CO c1(C(=O)NC2C3(CN(C(CSC(C)C)=O)C3)CC2)[nH]nc2ncccc12 C(C#CC(F)(F)F)NC(CCOCCN(C(Cc1c(C)ncs1)=O)C)=O N1(c2nccc(C(=O)OC)n2)CCC(C)(NC(c2ccnc(Cl)c2)=O)CC1 C1(NC(CN(C2CC2)CC)=O)CCCN(C(=O)CC2CCOC2=O)CCC1 c1(C(N2CCC(CC(=O)NCC(C(C)(C)O)O)C2)=O)ccc(F)c(Cl)c1 C1(NC(Cc2c(C)con2)=O)CC2CCC(C1C)N2C(=O)CC1(C)CCCO1 C1(c2cn(CCCO)nn2)(NC(C(SC)SC)=O)CCCOC1 N1(C(C(=O)NCC)=O)CCC2CCC(C1)N2C(=O)Cn1nc(C)c(Cl)c1C Cc1c(CNc2cccc(C(=O)NC3(c4ccccc4Cl)CC3)c2)cccc1O N1(C(CNC(CC)=O)=O)CC2CC2C1C(=O)NCC1CCOC1 CN1CCCCC1CC(N1C(CNC(c2csc(C(F)F)c2)=O)CC2CC12)=O c1(C(N(CC(CC)NC(C2(n3nccn3)CC2)=O)C)=O)cc(C)nc(O)c1 C1(C(=O)NCc2c(C(N(CC(F)Cl)C)=O)con2)C2CC3C(C2=O)C13 c1(OC)cc(OCC(=O)NCC23COC(C2)C(O)C3)cc(F)c1 Cc1nc(N)cnc1C(=O)NCC1CCN1C(=O)C=CC1CCC1 N1(C(C2CCN(Cc3ccc(C)o3)C2)=O)CCCC(O)(CO)C1 c1(C(C(=O)Nc2ccc(F)cc2)N(C2CCC2)CCC)ccc2c(c1)CCC2 c1(SC)cncc(NC(C2CC(C)N2C(=O)CC2CCC(C)(C)C2)=O)c1 CN1CCN(C(=O)C(O)(c2ccccc2)C2CCCC2)CC1 c1(C(=O)NCC(C)NC(C(CC)C)=O)cc(Cl)c(Br)c(OC)c1N c1(CN2CCC(NC(CC)=O)C2)cc(OC)c(C(=O)OCC)c(F)c1 N1(C(CCc2nc(=N)[nH][nH]2)=O)CCC2(CC2C(=O)NCCC(F)(F)Cl)C1 c1(N(C)C)ncccc1C(=O)NC(C)(C)CCNC(C1CCC(C(N)=O)C1)=O CCC(CC)C(C(=O)NC12CC1CN(C(C1(CC3CCC3)CC1)=O)C2)OC c1(OCCC)cccnc1C(=O)N(C)CCNC(C12CC(CCO1)C2)=O c1(C(=O)NCCCN(C(C(c2c(C)cccc2)C)=O)C)cncc(S(C)(=O)=O)c1 C(=O)(C1=NOC2COCC12)NC(C(C)O)C(=O)NCCOC(F)F C1(NC(CN(CCOC)C)=O)COC2(C1)CN(C(=O)C(C)(C)C(C)C)C2 N1(C(c2ccc(OC)nn2)=O)CCC2CCN(C(=O)CC3CS(=O)(=O)C3)CC12 c1(C(N(CCN(C(CC=CCC)=O)C(C)C)C)=O)cnn(C2CCCC2)c1C c12ccc(c(OC)c1)OC(CC)C(=O)N1C3CC1CN(C3)C2.C(COC)OC Cc1c(NCCCOc2cccc(Cl)c2)nc[nH]c1=NCC(C)N1CCOCC1 c1(OC)cc(NC(C2CC(C)CN(C(=O)Cn3nc(C)oc3=O)C2)=O)cc(F)c1 c1(CNC(C2SCCCS2)=O)cc(C(=O)NCc2ccncc2)n[nH]1 c1(C(=O)NCC2CC(OC)CN2C(C2COC2)=O)cn2cc(Cl)cc(Cl)c2n1 c1(CC)noc(C)c1CNC(=O)N(C1CC1)Cc1nnc(C)o1 CCC(C)C(C(=O)NC(Cc1ccco1)C(=O)NCC(CC)C(C)C)N(C)C N1(C(c2cc(CC(C)C)nn2C)=O)CCCC2(CCN(c3cc(O)ncn3)C2)C1 C1(NC(CCC=C(C)C)c2nnnn2C2CCOC2)COC(C)(C)C1 C(=O)(CC1OCc2ccccc21)NC(C)CNC(c1coc(CO)c1)=O c1(CC(=O)N(CC(C)N(C(CCCc2cc(C)no2)=O)C)C)c(C)noc1C N1(C(=O)NC(c2ccccc2)C=C(C)C)CCC12CCCOC2 C1(C2CCC2)(C(=O)NCC(CN(C(=O)CSc2ccc(O)cc2)C)(C)C)CCC1 C1(NC(C2C(C=C)C2)=O)CN(C(c2ncc(Cl)s2)=O)CCC12CCC2 N1(C(c2ccc(C#C)cc2)=O)CC(C)(C)CCC1CNC(=O)C(F)C1CC1 CC1(CC(=O)NC(c2cn(Cc3cnns3)nn2)(C)C)CCCC1 CC1CCCN(C(=O)C(=O)NC(C)C(=O)N(CCC#N)C)C1 N1(C(CCCC#CC)=O)CCC2CN(C(=O)CCC3CCCO3)CC12 C1(CNC(c2c(C)cc(O)nc2)=O)C(C2CC2)CCN1c1ncnc(C)c1F C(=O)(C#CC1(C)COC1)NC1CCN(C(COCCCCCC)=O)CC1C c1(-c2cn(CC(C)C)nc2)cc(C(=O)N(CC(F)(F)F)C)c2nccn2c1 c1(C(C)NCCCC2CCOC2)cnn(-c2ccccc2F)c1N C(=O)(C1Cc2ccccc21)N1CC(C2(NC(c3scc(C(N)=O)c3)=O)CC2)C1 N1(C(CCN(CCC)C)=O)CC(O)CC1CNC(C1CCN(CC2CC2)CC1)=O CC(C(=O)NCC12CC1CN(C(c1ncn(C)n1)=O)C2)C(C)(C)C Cc1cn(C)cc1C(=O)NC(C)(C)C=CC(=O)NCC1(O)CCN(C)C1 n1(C(C(=O)NC(C(C)C)C(=O)N(C2CCCCC2)C)C)c(=O)oc2ccccc12 C1(CNC(c2n(C)ncc2Cl)=O)CCCN(C(=O)CC2(C)CC2(Cl)Cl)CC1 c1(C(N(CC(CC)NC(=O)CC2CCC(=O)N2)C)=O)ccc(O)nc1Cl C(=O)(C(C)(C)CCCc1ccccc1)NCC(CNC(C1COC(=O)N1)=O)OC C1(CNC(C(N2CCNC2=O)C)=O)COCCN(C(=O)CCc2ccccc2)C1 Cc1ccc(F)c(CC(N2CCC(C(C)(C)NC(c3cc[nH]c(=N)n3)=O)C2)=O)c1 c1(C(=O)NCC23N(C(c4c(C)nccc4)=O)C(CC2)CC3)c(Cl)sc2nnsc12 C1(NC(N(C(C)Cc2ccccc2C)CC)=O)CC2(CCC2)C1OC n1(CC(N2CC(C(C)NC(=O)C(F)n3cccn3)C2)=O)nc2n(c1=O)CCOC2 c1(C(N2CCC(NC(c3cc(-c4cccnc4)[nH]n3)=O)C2)=O)ccc(O)cc1F Cn1cc(C(=O)NCc2cc(C(=O)NCC3(O)CCCOC3)co2)n(C)c1=O C1(CNC(c2cc(C)[nH]n2)=O)CC(C)CN(C(=O)CN2CCOCC2)C1 C1(C)(CC(N2CC(C)C(NC(c3cccc(N)c3)=O)C2)=O)CCCCCC1 C(C)(C(C)C(=O)NC1C=CC(C(=O)OC)C1)NC(c1cc(OCC)n[nH]1)=O c1(CC)nc(C(=O)NCC(C(C)C)NC(c2cc(CC(C)C)on2)=O)co1 C1(O)(CNC(C2(CCN(C)C)CCCC2)=O)CCN(C(=O)CCc2ccoc2)C1 c1(C(=O)NC2CN(C(C(C)CC3CCCC3)=O)CC2C)ccc(P(C)(C)=O)cc1 C12(C(=O)NCC#CCNC(c3cn(CC(C)C)nc3)=O)CCCCC1CCC2 c1(C(=O)NCCC(CNC(C(C)=C2CCCC2)=O)O)ccccc1C1CC1(F)F C1(NC(CCOC)=O)CN(C(=O)Cn2nccn2)CCC1(C)C.C12CC(C1)C2 c1(C(=O)NCC(CNC(=O)C=CC2CCCC2)OC)ccc(Br)cc1O CC1(CNC(c2cc(O)cc(O)n2)=O)CC(F)(F)CN1C(=O)CC1CC(=O)C1 C1(C#CC(=O)N2CCCC(CN(C(=O)C(F)(F)C(F)F)C)C2)(CC)CC1 N1(C(c2cccc(C)c2C)=O)CCCN(C(=O)CC(F)F)C(C)C1 C(C1c2ccccc2CN1C(c1cnc2[nH]cnc2c1)=O)NC(CCOCC)=O C(=O)(C(CO)C(C)(C)C)NCC1CN(C(Cc2ccc(C)cc2)=O)C1 N1(C(=O)Cc2ccc(Cl)c(Cl)c2)CCOC2(CCN(C(C3(O)CCC3)=O)C2)C1 N1(C(CC2(CCC#C)OCCO2)=O)CCCCC1CNC(=O)CC1CC2CC2C1 C1(C(C)C)N(C(=O)CC2CCCN(C(=O)CN(C)C(N)=O)C2)CC12CCCC2 CC(C)(C)C(CNC(c1cccc(C2CC2)n1)=O)NC(c1cnc(C2CC2)s1)=O C=C1CC(C(=O)NC(C)CNC(C2CCCN2CCC)=O)(Cc2ccccc2)C1 C12(C(=O)NCC3(O)CN(C(C4CC(C(F)(F)F)C4)=O)C3)CCCCCC1OCC2 O=C(N=c1ccn(CCCO)[nH]1)C1CCCCCN1C(c1cccc(F)c1)=O C(=O)(C1=CCCSC1)N1CCC(N2CCC(NC(C(CC)C#N)=O)CC2)C1 c1(C(=O)NC2(C)CC(NC(c3c(CC)noc3C)=O)C2)cccc(C=C(F)F)c1 Cc1cc(C(=O)NC2CC3CCC2(NC(=O)C(O)CC2CC2)C3)cc(O)n1 Cc1ccc(SCCC(=O)NCC2(c3cc[nH]n3)CC2)cc1 n1(C(C)C)cc(N(C(=O)CC2CCC(NC(=O)Cc3cccnc3)C2)C)cn1 c1(OCC(N2CC3C(NC(=O)COC(F)F)C(CC3)C2)=O)ccccc1[N+](=O)[O-] C1(C2CCN(C(c3ccc(Cl)c(C(F)(F)F)c3)=O)C2)(NC(C2C(C)(C)C2)=O)CC1 C(CN=C(NCC1CC1C1CC1)N1CCCC(N2CCCCC2)C1)OCCC=C N1(C(Cc2cccc(C(C)(C)C)c2)=O)CCC2(CC1)CN(C(C1CCO1)=O)C2 N1(C(=O)CCCc2ccsc2)CCCN(C(=O)COC(F)F)CC1CO C1(C(=O)NCC(C)(C)C(=O)NCCCn2cnnn2)CCCC12CCC2 Cc1cc(CN2CC(C)(CC(=O)Nc3cc(Br)ncc3C)C2)ccc1O CC(C)C(O)CC(=O)NC1CC(OCC(=O)NCC23CCC(CC2)O3)C1 c1(C(=O)NC(CN(C(=O)C=NOC)CC)C)cc([N+](=O)[O-])c(N)cc1F Cc1nc(NC(=O)CCNc2ccccn2)cc(N2CCC(N3CCC3)C2)n1 N#Cc1cnc(C(=O)NCCC2CCN(C(C3CCCCC3(F)F)=O)C2)c(Cl)c1 c1(OC)nccc2c(C(=O)NCC3CCN(C(=O)CCOC4CC4)CC3)c[nH]c12 N(C1=NCC2CCCC(C)N12)CC(C)Oc1ccc(C#N)cc1 C1(CCC(=O)NC(C2(C(N(CC(CC)OC)C)=O)CC2)C)NC(=O)NC1=O N1(C(c2cc(C)[nH]n2)=O)CC2CCCCC2(CNC(=O)CCc2ccccc2)C1 N1(C(C2CCC(=O)NC2)=O)CCC2C(C(=O)N(CCCCO)C3CC3)C2C1 C1(CNC(C2(CCC)CC(=O)C2)=O)CCCN(C(=O)C=Cc2cncs2)CC1 N1(C(C2(OCC)CCCCC2)=O)CCC(C)C(NC(c2cccc(C)c2)=O)C1 c1(OC)ncnc(C)c1C(N1CCC(N2CCN(C(C3CSC3)=O)CC2)CC1)=O C1(CNC(=O)COCCF)CN(C(c2cc(C(O)C(F)(F)F)ccn2)=O)CCO1 C(=O)(CCCCCF)N1CCC(N(C(C=CC(CC)C)=O)CCO)CC1 C12(NC(CC3(N(C(CCC(C)CN(C)C)=O)C)CC3)=O)CC1COC21CCC1 CC1CC(NC(c2nc(Cl)c(Cl)s2)=O)CCN1C(C1CNC(=O)N1)=O CS(=O)(=O)CCCC(=O)N1CCCC(CO)(NC(=O)CCN2CCC2)C1 c1(OC)cc(C)ccc1OC(c1cnccc1OCc1ncc(C(F)(F)F)[nH]1)=O c1(C(=O)NC(C2CCCCC2)CNC(c2cc(F)n[nH]2)=O)ccc2c(c1)OCC2 C(=O)(C(Cn1cncn1)NC(=O)C=Cc1ccco1)N(C1CCC1O)C C1(NC(C2CCN(C)C2=O)=O)CC2CC1CN(C(=O)C1=C(Cl)CCOC1)C2 C1(C(N(C)Cc2cc(C(C)C)on2)=O)CCCN(c2cc(C=O)ccn2)CC1 c1(C(=O)NCC2(OC)CN(C(C3CC(C(C)C)C3)=O)C2)cnc(N)c(N)c1 CC1CN(C(=O)C(=O)Nc2ccccc2I)CCN1S(C)(=O)=O CC1(C)C(C(=O)NCC2CCCCC2)CCN1C(C1CC(F)(CF)C1)=O N1(C(C(c2cn(CC)nc2)=O)=O)CCN(C(c2cccc(F)c2Cl)=O)CCC1C Cc1cc(CCC(=O)NCC2CC2NC(c2c[nH]cc2C)=O)c(C)s1 N1(C(CC2(NC(CCCOCC=C)=O)CC2)=O)CCC(=O)N(C)CC1 N1(C(CCCNC(=O)OC)=O)CC2(CC(NC(=O)Cc3cc(Cl)ccc3Cl)C2)C1 c1(CNC(C(=O)NC2CC(NC(C)=O)CC2n2ccnn2)=O)cccc(O)c1F C1(NC(CC)=O)CC2CC1CN(C(c1c[nH]c(C(N)=O)c1)=O)C2 C1(CCNC(C2CN(C)C2)=O)CCCCN1C(=O)Cn1cc(CO)nn1 C12(NC(C3CCCCCC3)=O)CCN(C(=O)C=CC=C(Cl)Cl)CC1C2 n1(C(CC)C)ncc(C(=O)NC2COCCC2NC(c2ccncc2O)=O)c1C C1(NC(CN(CC)CC)=O)C2CCC1CN(C(C1CC3(CC3)CO1)=O)C2 N1(C(c2cc3cccc(C)c3[nH]2)=O)CCCC(C2CN(CCF)C2)C1 c1(NC(C2C(C(N(CCN=[N+]=[N-])CCO)=O)C2)=O)cnc(-c2ccco2)[nH]1 C1(NC(c2ccc(C(N)=O)s2)=O)(CO)CCCN(C(=O)C(F)(F)CC2CC2)C1 CC1(C(=O)NCc2csc(C(N3CCN(CC(N)=O)CC3)=O)c2)CC2CC2C1 C(CC(CC)C(=O)NCCCNC(=O)C(C)NC(c1cc(F)cc(F)c1)=O)=CC C1(CNC(CCC)=O)CC12CCN(C(=O)Cc1ccc(C(F)(F)F)nc1)CC2 c1(OC(C)C)ccc(C(=O)N(C)CCN(C(=O)C(C)CC(N)=O)C)cc1N Cc1cc(Cl)ccc1OCC(N1CCC(NC(=O)C2=CCC2)C(C(C)C)C1)=O CC(F)(F)CCC(=O)NCc1ccc(C(=O)NCc2nccn2C2CC2)o1 C=CCN=c1[nH]c(C(N2CC3(CCCC3NC(C3CC4CCC3C4)=O)C2)=O)cs1 c1(CN(C(=O)CCC2CCCN2C(c2ccoc2Cl)=O)C)cccc(F)c1 Cc1cnc(CNC(C2CC23CCN(C(=O)Cn2ncnn2)C3)=O)c(C)c1 c1(OC)ccc(OC)c(C2CN(C(=O)N(CC(C)(C)N(C)C)C)CCO2)c1 N1(C(c2ncccc2Cl)=O)CCC2(CC1)CN(C(C1CC13CC3(F)F)=O)C2 c1(C(=O)NC)cccc(NC(=O)CC2CN(S(=O)(=O)CC#N)CCO2)c1 C1(C(N(C)CC2CCNCC2)=O)C2CN(S(=O)(=O)CCC3CCS(=O)(=O)C3)CC12 C12(OC)CCC(C(=O)NCC3(O)CCN(C(c4nnn(CO)c4C)=O)C3)(CC1)C2 c1(C(=O)NC2CCC(C(N3CC=C(COC)CC3)=O)CC2)ccn2ccccc12 C(=O)(CC(C)CCC)NC1C(C(=O)NCC2(C#C)CCC2)CCOC1 CC1CC(F)(F)CCN1C(C1(CCNC(=O)COCC2CCCC2)CCCC1)=O N1(C(c2cc(C)[nH]n2)=O)CC2CC1(c1cn(Cc3ccc(C(=O)O)o3)nn1)CO2 c1(C(=O)NC(C)CCC(=O)NCC2(C)CCCC2O)cccc(F)c1N c1(C(N(C)CC2CN(C(C(C)C3CCCO3)=O)C2)=O)cccc(=S)n1O C1(OCC(N)=O)CCN(C(=O)CC2CCN(C(=O)C(F)n3ccnc3)C2)C1 C1(C(=O)NC(C2C(C(=O)OC)C2)C)CC(NC(C2CNC(=O)O2)=O)CCO1 c1(C(N(C2CCC(NC(C3(OCC)CCC3)=O)C2)C)=O)ncccc1F C1(CC#C)(C(=O)NCC(c2ccco2)O)CCCCN1 O=C(C1=NOCC1)NC1CCCC(NC(c2cc(C(F)(F)F)ns2)=O)C1 C1(C)(CNC(CCOC)=O)COCCN(C(=O)CC2CN3CCC2CC3)C1 C(=O)(CC(C)(C)C(F)F)NCCC(CNC(c1ncc(C)cc1F)=O)O C1(CC(=O)N(CCC(=O)NCCCN(C)C)CC=C)C=NN(C)C1=O N1(C(c2nc(C)oc2)=O)CC(C)CN(C(c2ccc3c(c2)COB3O)=O)CC1C Cc1ccc(C=CC(=O)NC2CCC(CNC(=O)CCC3CCC3)CC2)s1 Cc1ccccc1N=c1[nH]c(COC(=O)CC2CCc3ccccc32)nc(=N)[nH]1 C1(N(C2CCN2C(C)(C)C)C(C)=O)C=CCN(C(C2CCS(=O)CC2)=O)C1 C1(CNC(C=C(C)C)=O)(CNC(=O)OC(C)(C)C)CCCN1C(C1C=CCC1)=O C(=O)(C(=O)N=c1cc(C)o[nH]1)NCC1N(C(c2c(OC)c(C)ncn2)=O)CCC1 O=C(C1=NOC2(CCC2)C1)NC1CCCC(CO)C1 C1(NC(CCC#C)=O)CCN(C2CCN(C(C3(CC(C)C)CCC3)=O)C2)CC1 c1(C(N2CCC(NC(C(CC)CC)=O)C2)=O)cc(=O)oc2ccc(O)cc12 N1(C(C2(C)CCCCCC2)=O)C2CCC1C1CC1(NC(=O)CC1(CO)CC1)C2 c1(OC)cc(C(=O)NC(C)C(C)NC(C23CC(C)(CCO2)C3)=O)cnc1O CN1CCC(C(N2CC(C(N)=O)(CNC(c3n[nH]c(C(C)(C)C)n3)=O)C2)=O)C1=O Cn1ccc2cc(C(N3CC4CC(C3)N4C(=O)C(F)Br)=O)ccc12 c1(C(=O)NC(CNC(C(COC)N(C)C)=O)C)cc(Cl)nnc1O N1(C(Cc2cc(C)[nH]n2)=O)CC2CCCC(NC(=O)CN3CSCCSC3)C2C1 C1(NC(c2c[nH]c(Br)c2)=O)CN(C(c2cc(-n3cccn3)ccn2)=O)CC1F C1(C(=O)NCC(C)CC(=O)NCC2CC2(C)C)CC2(CCO1)CC2 C=C(C)CC(C(=O)N1CCC(NC(c2[nH]nc(C(F)(F)F)c2C)=O)C1)NC(C)=O c1(CC)c(C(=O)NCC2(O)CCN(C(C3CC4CCC3CC4)=O)C2)cccc1F S(=O)(=O)(c1cnn2ccc(N3Cc4ccccc4C(C)(C)C3)nc12)NCC(C)O c1(C(=O)OC)c(C)[nH]c(C(=O)C(C)OC(=O)CC23COC(CF)(C2)C3)c1C C(=O)(C1=COCCC1)NCCNC(=O)Nc1n(C(=O)OCC)ncc1 N1(C(C(CO)NC(C(C)C)=O)=O)CCC2CN(C(C3CN4CCN3CC4)=O)C2C1 n1(C(CC)CC)ncc(C(=O)NC(C)CCNC(=O)C=CCCC(C)C)c1C C1(C(=O)NC(C)CCNC(=O)CC2CCOCC2)CCc2ncc(Br)n2C1 CC1=NOC(C(=O)N(C2CCN(C(=O)Cc3csc(-c4ccco4)n3)C2)C)C1C C(C(C)(O)C(C)(C)C)NC(CCC1CC(NC(C(C)N=[N+]=[N-])=O)C1)=O C(C)(CNC(=O)C(CO)NC(N)=O)(C(C)C)NC(Cc1cc(C)on1)=O O=C1COC(C(=O)NCC2CN(C(=O)Cn3ccsc3=N)C2)C1 C(=O)(C(CC(C)C)NC(=O)CC(F)(F)F)N(CCN(C(CC(=O)OCC)=O)C)C N1(C(C)=O)CCCC(C2CN(Cc3ccc(Br)c(C(F)(F)F)c3)C2)C1 C=CCC(CNC(=O)CC1COCC1O)NC(=O)Cn1nnc(-c2cccs2)n1 C(CN1C(=O)C(C)Oc2ccccc21)NC(C(c1cn(CC)nc1)=O)=O Cc1cccc(N)c1C(N1CCCC(NC(c2c(Br)cnn2C)=O)C1)=O C(=O)(C(C)C(O)CC(C)C)N1CCC(C(C(=O)NC(CCOC)(C)C)F)C1 N1(C(C(C=C)CC)=O)CC(C)CN(C(=O)CCCCC2CC2)CC1C N1(C(c2c(C(=O)OC)cccc2)=O)CCC(F)(F)C(CNC(=O)C(C)N(C)C)C1 C(=O)(C(CC(C)C)C(C)C)NC(CCC(=O)NCCC(CC)(O)CC)(C)C C=Cc1ccc(C(=O)N(C)CC2CCN(C(C3CCN3S(C)(=O)=O)=O)C2)cc1 c1(C(=O)NC2CN(C(c3cnc(N(C)C)s3)=O)CC2C(F)F)ccc(F)c(N)c1 c1(C(=O)OC)nc(C(=O)NC2CC(CCNC(C3(Cl)CC3(F)F)=O)C2)cs1 C1(C)(CC)C=C(C(=O)N2CCCC(F)(C(=O)NCc3nc(C)cc(O)n3)C2)C1 C(=O)(C(C(F)(F)F)C(F)(F)F)NC1CC(NC(CNC(c2cc(C)nn2C)=O)=O)C1 C(=O)(C(CC(C)C)NC(c1csc(CNC(=O)CCn2ccc(C)n2)c1)=O)NC N1(C(C2(OC)CCCOC2)=O)CC2(CCC(NC(=O)CSCCC(C)C)CC2)C1 c1(NCCC(=O)NC)[nH]c(=NC2COC3(CCCC3)C2)nc2c1ncn2C(C)C C1(C(=O)NCC(CNC(C23CC(C)(C2)C3)=O)OC)CC(=O)N(CC(C)C)C1 C123COC(C1)(C2)C3.Cc1nnsc1C(=O)NC(CNC(C1CCN(C)C1)=O)C1CC1 Cc1nccn1C(C)C(=O)N(C(C)C(=O)NCCCC(F)F)C C1(NC(=O)CC=C(Cl)Cl)CC(NC(c2ccc(Br)cc2)=O)C12CCC2 C=CC1CN(C(C2CN(C(=O)CCC#CC)CCN2C)=O)CC1O C1(NC(CCC#C)=O)CCC2(CC1)CC(NC(=O)C(C)C(F)(F)C(F)F)C2 c1(C(=O)NC(CC=C)CNC(=O)CC(C)N(C)C)cc2c(F)cc(F)cc2[nH]1 N1(C(C2CC(C)OC2)=O)CCC2(CC1)COC(CNC(c1ccc(=O)oc1)=O)C2 C12(C(=O)NC3CCN(C(C(C=CCCC)O)=O)CC3)CCC(C(F)F)(CC1)CC2 C12(CNC(N(c3ccc(C(F)(F)F)cn3)C)=O)CC=CCN1CCC2 c1(C(N2CC(NC(CCC(C)(F)F)=O)C2)=O)cc(C(F)(F)F)ncc1[N+](=O)[O-] c1(C(=O)NC2CN(C(C=C(C)c3cccs3)=O)C3C2C3)c(C)cccc1F c1(N2CCC(CNC(C3(C)CCC(C)C3)=O)C2)ncccc1C#N C1(NC(c2n(CC)ncc2)=O)CCCC12CN(C(=O)CC1(CO)CCCC1)C2 c1(C(N(CC(C)NC(C(CC)OCC)=O)C)=O)cnc2ccncc2c1 C=C1CCC(C(=O)NC2CN(C(=O)C=CC(=O)NC3CC3)CC2O)CC1 c1(C(N2CC(NC(C(CC)C3CCOCC3)=O)C2)=O)[nH]c(O)nc1C N1(C(CCc2ccc(=N)[nH]c2)=O)CCCCC(CNC(c2nc(Cl)c(Cl)s2)=O)C1 CCC1=NOC(CC(=O)NCC(CNC(=O)CCc2ccc(Cl)cc2)CO)C1 C1(C(=O)NCCC2CCCC3CC23)CC2(CCC2)CN1C(=O)C(O)C(F)(F)F c1(C(=O)NCCCN(C(C2(C(=O)OCC)CC2)=O)C)nccc2c(F)cccc12 c1(C(=O)OC)ccc(S(=O)(=O)N2CCC(NS(=O)(=O)CCc3ccccc3)C2)n1C N1(C(C=NOC)=O)CCC2(NC(C3CCN(C4CC4)CC3)=O)CCCCCC12 C1(CNC(C2(OC)CCCOC2)=O)CN(C(C2CSCC(=O)N2)=O)CCC1C C1(F)(CNC(C2C(CC)C2)=O)CCN(C(c2c(Cl)nsc2Cl)=O)CC1 CC(C)(CCCC(=O)NC1CC1F)NC(C1CC(C2CC2)=NO1)=O O(S(=O)(=O)c1ccc(C(C)(C)C)nc1)c1ccc(OCCCC)cc1 C=CCC(Cc1ccccc1)C(=O)NCC(C1CC1)NC(C1(CO)CCCC1)=O Cc1cc(NCC2CC(F)(F)CO2)ncc1S(=O)(=O)NC(C)(C)CF c1(Cn2c(C(C3CCOC3)Nc3cn(COC)nc3)nnn2)ccc(OC)cc1 C1(O)(C(C)NC(=O)C(c2ccccc2)O)CCN(C(=O)CCC(F)(F)F)CC1 c1(OC)c(C(=O)NCC=CCNC(C2(C)CC=CCC2)=O)cccc1Br C1(O)(CN(C(C2N(CC)CCCC2)=O)C)CCN(C(c2nc(O)c(C)s2)=O)CC1 c1(NC2(c3nnnn3C(C)C)C(OCC)CCC2)cc(C)c2nccn2c1 C(C(CC(F)(F)F)NC(=O)C(C)NS(C)(=O)=O)NC(CC1(OCC)CC1)=O N1(C(CN2C(C)CCC2)=O)CCCN(C(=O)CN(C(=O)OC(C)(C)C)C(C)C)CC1 c1(CC(=O)NC2CCN(C(c3c(CC)[nH]cc3)=O)CC2)ccc(C)c(Cl)c1 c1(C(N(C2CCN(C(c3csc(C(C)(F)F)n3)=O)C2)CCC)=O)ncccc1N c1(OC)ccc(-c2cncnc2CN2CCCC2c2c(C)n[nH]c2C)c(F)c1 c1(CC2OCC(CNCC3(OC)CCCC3)C2)cc2nnc(C(C)(C)C)n2cn1 CCCCC(C)CCC(=O)N1CC(NC(c2cnn3c2CCCC3)=O)C(OC)C1 N1(CCNC(c2cnc(Cl)[nH]2)=O)CCN(C(C2CCOC2C(F)(F)F)=O)CC1 c1(C(N2C(CN(C(=O)C#CC(C)C)CC)CCC2)=O)cc(S(N)(=O)=O)ccc1O CCCC(C(O)C(=O)N1C2CCC1(CO)CC2)NC(c1nnn(C)c1CC)=O N1(C(c2nc(C)oc2)=O)CCCN(C(C2CC2C)=O)CC1C(C)C CC1CCCCC1C(N1CCN(C(C)CNC(=O)C(F)F)CC1)=O C(=O)(C1=CCCCC1)NC1CC(C)(NC(CC2(C)CC2F)=O)C1 C(=O)(C1=C(C)CCCC1)N1C(C)CC(NC(Cc2ccc(OC)cc2C)=O)C1 N1(C(c2c(C)ocn2)=O)CC(F)CC1C(=O)NCCCc1cccnc1 c1(C(N2CCN(CC(=O)NC(C#C)C(C)(C)C)CC2)=O)cccc(F)c1F CC(CC(C)NC(=O)C=Cc1cn[nH]c1)NC(=O)C(C)(C)Nc1ccccc1 c1(C(=O)NCCC(C)NC(C2C(OC)(OC)CC2)=O)ccc2c(c1)CCO2 CC1CCN(C(C2(CCN(C)C)CC2)=O)CC1N(C)C(c1cnnc(O)c1)=O c1(C(=O)NCC2N(C(C3OCC(C)C3)=O)CCC2)cc(O)cc(Br)c1 c1(C(=O)NC2CC(F)(F)CC2O)cc2cc(F)c(F)cc2[nH]1 C1(C(=O)NCCC2(NC(CCCC(N)=O)=O)CCC2)Cc2ccc(F)cc2O1 N1(C(CC(=C=C)C)=O)CC2(CNC(C3CC4(CC4)CO3)=O)CC1CO2 N1(C(C(C)NC(C)=O)=O)CCCC12CCN(S(=O)(=O)c1cc(Cl)ccc1Cl)CC2 CC(C(C)(C)C(=O)NC1COCCN(C)C1)NC(=O)C=Cc1cc[nH]c1 CC(C)C(O)CC(=O)NC1CN(C(c2ccnn2CCN(C)C)=O)CC1C c1(C(=O)NC(CCC)CCCNC(=O)C(F)n2cccn2)cc(F)c(F)cc1O c1(C(=O)NCCCCC(C)NC(c2n[nH]c(C)c2O)=O)cc2n(n1)CCN(C)C2 C(C)(C(C(C)C)NC(=O)C=CC1CCCCC1)NC(COc1cc(C)on1)=O c1(C(=O)NC(CNC(C(C=C)OC)=O)(CC)CC)ccc(OC)c(N)n1 C(CCN=c1[nH]nco1)N(C(c1cccc(OCC(C)C)n1)=O)C Cc1cn(C)cc1C(=O)NC(C)(C)CNC(=O)C(c1ccc(CC(C)C)cc1)C C1(C)(CC(=O)N(CCN(C(=O)C(C)n2cnnn2)C(C)C)C)CC1(F)Cl Cc1noc(Cl)c1CCC(=O)NC(C)C(C(C)C)NC(c1ccsc1C#N)=O Cc1ccc(C2(C(=O)NCC(C)NC(=O)CCC(C)(C)C)CC2)cc1Cl c1(C(C(=O)NCC=C)N(C(c2cccc(C)c2)C(C)C)C)ccc(OC)cc1 c1(C(N2CCC(O)(CNC(C3CC34CC4)=O)C2)=O)cc2c(s1)CCCCCC2 S(=O)(=O)(c1cc(C(=O)NC2CCN(C(c3ccc([N+](=O)[O-])cc3)=O)C2)co1)NC C12(CNC(CN(C3CC3)CC)=O)CC(CN1c1ncns1)C2 c1(N(C)C)n[nH]c(C(=O)NC2CCC2C(=O)NC(=O)COc2ccccc2)n1 c1(COCC(=O)NCCN(C(=O)Cc2nnc(C)s2)CC)cccc[n+]1[O-] C(C)(CO)(C(=O)NCc1cc[nH]c1C(=O)N(C)CCc1ccncc1)OC C1(CNC(C(C)O)=O)(NC(=O)COC2CCCCC2)CC=CC1 c1(C(=O)NC2CC3CN(C(c4nc(OC)oc4)=O)C2C3)ccc2c(c1)COC2 CC(C)CCC(O)C(=O)NCC(CNC(c1ccc(C(=O)N(C)C)cc1)=O)CO c1(C(=O)NC(C2CN(C(C3(C)CCCC3)=O)C2)C)cc(N2CCCC2)ncn1 c1(C(N2CC(F)CC(NCc3nc(C(C)C)sc3)C2)=O)cc2cc(Br)ccn2n1 C1(C(=O)NCC=CCOC)C2CC3C(C2NC(C2CC2C(N)=O)=O)C13 c1(SC)cccc(C(=O)NCC(C)N(C)C(C2CCC(C(C)(C)O)CC2)=O)c1 c1(OCC)ccccc1OCC(=O)NC1CCC1NC(C1CC2C=CC1O2)=O c1(C(N2CCN(C(C(C=CC)O)=O)CC2CF)=O)coc(S(=O)(=O)NC)c1 c1(C(N2CCN(C(C3C(=C)C3)=O)CC2C)=O)ccc(S(N)(=O)=O)cc1Cl Cc1ccc(F)c(C(=O)NC2C3CC2N(C(c2cc(C4CCC4)nn2C)=O)C3)n1 Cc1cc(C(N2CCN(C(=O)Cc3ccnnc3O)CC2C)=O)c(C)n1C C12(NC(C(C=C)OC)=O)COC(C1)C(NC(c1sccc1C(C)C)=O)C2 S(=O)(=O)(c1ccc(F)cc1)N1C(CNC(c2cc(Br)cs2)=O)COCC1 c1(CCC(=O)N(C2CC(=O)N(C)C2=O)CCC)ccc(F)cc1F N1(C(C(C=C)C)=O)CC2(CCCC2CC(N2CCn3nccc3C2)=O)C1 C1(C(N(CC(C)O)C)=O)CN(C(c2ccn(CCF)n2)=O)CC12CC2 Cc1cc(Br)c(F)cc1NC(=O)NC(CO)C(O)c1ccccn1 C1(OC(C)(C)C)CC(F)CN(c2nnc(-c3ccc(Br)s3)n2CC2CC2Br)C1 n1(CC)cc(C(O)CNC(=O)C(=O)NC2CC2)cn1 c1(NCC)ccc(Cl)cc1C(=O)NC1CCCC1NC(=O)CCCCC#N C1(O)(CNC(CNC(CC)=O)=O)CCCN(C(=O)CCOC2COC2)CC1 N1(C(CCCC#C)=O)CC(C)CN(C(=O)CCc2cnco2)CC1C Cc1cc(C)n(CC(N2CC3C(NC(=O)C(C(C)C)N(C)C)C3C2)=O)c(=O)n1 C(=O)(C1CCCc2cncn21)N1CC2(CCN(C(CC(C=C)CC)=O)C2)C1 S(=O)(=O)(c1ccc(C#N)c(NCc2nc(Cl)cs2)c1)N1CCCC(C=C)C1 CC(CN=c1nc2scnc2c(NCC(C)(F)F)[nH]1)C(C)(F)F N1(C(C2(c3ccccc3)CCN(C)C2)=O)CCN(C(=O)CC2(C)CC2)C(CO)C1 Cc1ccnc(C(=O)NC2(CNC(=O)CC(C)(C)C3CC3)CCCC2)c1F C(=O)(CCC1=NNC(=O)CC1)NC.C12(C)CCCCN1C(=O)NC2=O.C(C)(C)(C)NCC CC(C)(C)C(=O)C(=O)NC1CN(C(c2c(O)cccc2Cl)=O)CCC1C(F)(F)F Cn1ncc2ccc(C(N3CC(NC(=O)CC4(O)CCOCC4)C(F)C3)=O)cc12 c1(C2(COC(CC(Cc3cccc(OC)c3)C)=O)CC2)cc(F)ccc1F C1(O)(CNC(=O)C(O)C2CCC2)CCN(C(C2CC2(Br)Br)=O)CC1 Nc1ncc(C(=O)NCCC(=O)Nc2ccccc2CO)cc1Br C1(CCNC(=O)NC2CC2)CN(C(C2CCC3CC2C3)=O)CCCO1 C1(NC(=O)C=C2CCC2)CCCN(C(c2ccncc2)=O)CC1F C1(CN(C)C(C2CCC(O)C2)=O)CCCN1C(=O)CN1CC(F)(F)C1 C1(C(=O)NC2CCN(C)C(=O)C2)C(C2CC2)CCN1C(=O)CCC(N)=O C1(C(N(CCNC(C(C)SCCCC)=O)CCC)=O)CCC1(OC)OC Cc1sc(N)c(C(=O)NC(CNC(=O)C=Cc2cccc(CO)c2)C(C)C)c1C c1(C(=O)NCc2c(CCNC(c3n(C)cnc3)=O)ocn2)ccc([N+](=O)[O-])cc1 N1(CC(=O)N(CC(N)=O)C)CCC(N2CC=CC2)C1 c1(C(=O)NCc2cc(O)ns2)ccc2c(=O)cc[nH]c2c1 c1(-c2noc(C)c2C(N2CCC(=O)NC2=O)=O)cccc(S(C)(=O)=O)c1 C1(CN(C(=O)CS(N)(=O)=O)C)CCCN(C(C2CCS(=O)(=O)C2)=O)C1 C(=O)(CCCC(F)F)N1CC(NC(C2(C)C=CCC2)=O)C(c2ccccc2)C1 C1(CNC(C(CC)(C)OC)=O)Cc2ccccc2CN1C(C1CC(SC)C1)=O N1(C(C(C)NC(C)=O)=O)CC=CC1C(N1CC(CN=[N+]=[N-])C1)=O C(=O)(C1=NNC(=O)CC1)NC(C1CCCN1C(C1OCC1(C)C)=O)C c1(OC)ccc(C(=O)NC2(CCCNC(=O)C(F)CC(C)C)CC2)c(O)c1 c1(NCC2CN(C(C(CC)OC)=O)C(C)C2)nc(Cl)nc(CC)c1C#N C(=O)(CCC(=O)C(C)(C)C)N(CCC(=O)OCC)Cc1ccccc1 C12(C(=O)NCCC(C)NC(C3C4CCC3CC4)=O)CCCC1CC(=O)C2 CC(CCCNC(=O)CC1(O)CCCC1)NC(C1(C2CC2)CCCO1)=O CCCC(CCCO)C(=O)NCCOC1CN(C(C2CCCCC2(C)C)=O)C1 N1(C(CC(C)F)=O)CCN(C(=O)Cc2cccnc2O)CC1c1ccccn1 CCCS(=O)(=O)C(C)C(=O)NCC1CC2(CC2)CN1C(=O)CNC(=O)CN(C)C C12(CC(=O)Nc3nonc3N)CCC1CN(C(=O)C=CCC(=O)N1CCCC1)C2 CC1(C)CC(NC(C2(C)CCCN(C(C3CC(=O)CCO3)=O)C2)=O)CCO1 N1(C(c2c(CNC(C(C)OCC)=O)cco2)=O)CCS(=O)C(C)C1 CC#Cc1cncc(-c2csc(-c3nccn3C3CCCC(C)C3)c2)c1 C#CC1CN(C(=O)CC2CCCCC2)CCN1C(c1cc2nccnc2[nH]1)=O n1(CCCC)cc(C(=O)NCC2CC2NC(=O)CC2(NC(C)=O)CC2)nn1 c1(C(N2C(Cn3cc(C(COC)(C)O)nn3)CCCC2)=O)c[nH]nc1S(N)(=O)=O N1(C(C(CCCC)C)=O)CCC2(CC1)CC(NC(c1cc(Cl)cnc1Cl)=O)CO2 c1(C(=O)NCc2c(C(N(CC(C)CO)C)=O)cco2)cccc2c1CCC2 C1(CC)(CC)CN(c2cc(NCc3c(Br)nnn3C)ncn2)CCS1=O c1(C(N2C3CN(C(CC4CCN(C)CC4)=O)C(C3)C2)=O)nccc2ccccc12 c1(C(=O)NC2CCC(C)(CNC(c3c(C)csn3)=O)C2)cc(C)c(C)nc1C c1(C(=O)NCCN(C(C2C=CCCC2)=O)CC2CC2)ccc2nn[nH]c2c1 N1(CC(=O)N(C(c2ccccc2)C)C)CCC(NC(=O)CC2CC2C)CC1C c1(C(=O)NC2(CNC(C3(C)CC3(Cl)Cl)=O)CC2)nn(C(F)F)cc1Cl N1(C(C(CC)NC(N)=O)=O)CC2(CCN2C(C2CCCC2C(F)(F)F)=O)C1 c1(N2CCC(CC=C)(NC(c3cc(OC)ns3)=O)CC2)ncc(C#N)cc1F Cn1ccc2cc(CN(c3nc(C)ncc3Br)C3CCCCNC3)ccc12 N1(C(CC(=O)NCC)=O)CC2C(CNC(c3cccnc3CO)=O)C2C1 n1(C2CN(C(c3coc(C4CC4)n3)=O)C2)cc(CNCC2(O)CCSC2)nn1 c1(OC)ccc(F)cc1C(=O)N(CCC1(O)CCCN(S(=O)(=O)CCCl)C1)CCN N1(C(CC(C(F)F)NC(C2(C(C)=O)CC2)=O)=O)CCOCC(C)(F)C1 c1(C(=O)NC2CC(NC(c3cc(Cl)c(Br)[nH]3)=O)C2)cccc2c1CCOC2 CC(C)(Cn1cc(CC2CCCC2)nn1)CC(F)F c1(C(N(CCN(C(=O)CC(C)F)CC)CC)=O)ccc(O)c(C(C)C)c1 CCC(C)(CO)C(=O)OCCCc1ccsc1C(=O)OC CC1(Br)CC1C(=O)N(CCCNC(=O)CSc1cccs1)C1CC1 C(=O)(CCCC(F)F)N1C(C2(NC(=O)CCc3cnccn3)CC2)CCC1 C(=O)(CC1OCCc2sccc21)N1C(CNC(c2cccc(C)c2F)=O)CC1 c1(C(=O)NCC2(O)CCN(C(C(CCSC)N(C)C)=O)C2)cc(F)c(C)cc1F c1(C(=O)NC2(CO)CN(C(CC(=C=C)C)=O)C2)cnc(C)nc1OC C1(C(=O)NCC(CC)N(C(=O)CC2CN3CCC2CC3)C)CC1C1CCCC1 c1(C(N(C2C(C)CN(C(C3CCCCC3)=O)CC2)C)=O)ncc2n1CCCC2 C1(NC(C(C)Oc2ccccn2)=O)CC2CCC(C1C)N2C(C1SCCS1)=O C1(C)(CNC(CC2C(C)(C)CC2)=O)CCN(C(c2c[nH]nc2C2CCCO2)=O)C1 C(CS(=O)(=O)CC(=O)NC(C(N1CCC(OCCO)C1)=O)C1CC1)OC c1(C(=O)NC2CC(C)(NC(C(n3cc(Cl)cn3)C)=O)C2)ccc2snnc2c1 c1(OC)nn(C)cc1C(=O)NC(CC1CC1)CC(=O)N1CCC(c2ncco2)C1 c1(C2CCN(C(=O)Nc3c(CN(C)C)cccc3)CC2)nnc2cnccn12 CCCCCCCC(=O)N1CCCC(N(C(=O)CC(C)c2cnn(C)c2)CC)C1 C1(C(=O)OC)CC2(CCCC2)CCN1C(=O)C(=O)NCc1cnn(CC(F)F)c1 C(CCC(=O)N1CC(O)(CN(C(=O)COC2CCOCC2)C)C1)OCCOC C1(F)(C(=O)Nc2c(N(C)C)cccc2)CCCN(C(c2cc(C(N)=O)[nH]n2)=O)C1 C(N=c1[nH]c(-c2ccccc2)nc(=NCC=C(Cl)Cl)[nH]1)c1cc(O)nc(O)n1 N1(C(C2N(CC)CCC2)=O)CC(CO)C2(C1)CN(C(c1cc(C(C)=O)c[nH]1)=O)C2 c1(C(N2CCC(C)(NC(C(C)SCC)=O)C2)=O)cc(C)c(C)c(F)c1 c1(C(=O)NCC(C)N(C(C2CC2(C)C)=O)CC)ccc2cccc(OC)c2n1 C1(NC(CCN(C)CC)=O)CC2(C1)CC2NC(C1C(C#N)C1(C)C)=O c1(OC)ccc2c(n1)NC(C(=O)NC1CCCCN(C(C3CC=CCC3)=O)C1)C2 C1(C(=O)NC(c2nc(C)[nH]n2)C)CCN(C(c2ccc(CC#N)cc2)=O)C12CC2 C1(C(=O)NCC(COC)NC(c2n[nH]cc2Cl)=O)CCC(OC)CC1 N1(C(c2c(C)noc2)=O)CCC(C2CC2)(CNC(=O)C=Cc2cnccn2)C1 n1(NC(CCOC)(C)c2nnnn2C(C)C)cc(C)ccc1=O CC1=C(C(=O)NC2CCCC2NC(c2cc(CCO)on2)=O)CC1 C1(C)(C(=O)NCC2N(C(c3c(N)ccc(CCC)c3)=O)CC2)CC(C(C)C)=NO1 C1(CNC(COCCCC)=O)(NC(c2ccnn2C(C)C)=O)CCCCCC1 N#Cc1c(Cl)nsc1NC(CNC(c1cnc(Cl)c(C2CC2)c1)=O)CO Cc1cc(N2CCCC2CNC(=O)CCc2nccs2)c(Br)cc1[N+](=O)[O-] c1(C(=O)NC(C(=O)N(CCC(=O)OCC)C)Cn2ccnn2)ccccc1O c1(COC(C2CC3CC(N(C)C)C3C2)=O)c(-c2ccc(F)cc2)cc(F)cc1F C1(C)(OC)CCCN(C(=O)CCC(C)NC(=O)CN(C)C)C1 Cc1ccc(C2(C(=O)NC3CCN(C(=O)CCC4CC4)C3C3CC3)CC2)c(F)c1 n1(CCC(=O)NC(CNC(C2N(C)CCC2)=O)C2CCC2)ccc2ccccc12 c1(C(N(CC(O)CN(c2cc(O)nc(COC)n2)C)C)=O)cnc2ncccn12 N1(C(c2scc(CNC(COC(C)=O)=O)c2)=O)CCC2(CCOCC2)C1 C1(CNC(CNC(C)=O)=O)CCCN(C(c2cccc(C3CNC(=O)C3)c2)=O)C1 C12(C(N3CC(CCNC(CC4CCC(C)CC4)=O)C3)=O)CCC(C(F)F)(CC1)C2 c1(C(=O)OCC)cc(NC(=O)NCC2(CO)CC=CC2)cc(COC)c1 N1(C(c2coc(C(F)(F)F)n2)=O)CCC(n2cncn2)CC1 C1(COC)(CNC(C2CC(CF)C2)=O)CCN(C(=O)Cc2ncsc2Cl)C1 CC1(C)CCN(C(C2(c3ccccc3Cl)CC2)=O)CC1NC(C1CC1C1CC1)=O C(CCOC)(C(=O)N1CCC(C(=O)OCC)O1)NC(CCCCC)=O C1(CN(C)C(c2cccc(CO)c2)=O)CCCN(C(=O)CC2CC(O)C2(C)C)C1 c1(CC)nc(CC(=O)NC(C)CCNC(c2ncoc2C2CCCO2)=O)cs1 N1(Cc2c(OCC)cccc2)CCCC(F)(CNC(c2coc(C(C)C)n2)=O)C1 N1(CCC)CC(NC(N2CCC(CCc3ccccc3)CC2)=O)CC1=O c1(C(N2C(CNC(CC(C)c3ccco3)=O)CC2)=O)cccc2c(C#N)c[nH]c12 C1(=O)C(C(C)C)N1.CCCCC(=O)NC1CCC(CN(C(C)=O)CC)C1 N1(C(CCNC(C)=O)=O)CCCC(C(C)NC(c2csc(-c3ccco3)n2)=O)C1 C(=O)(CCCCCC#N)N1CCC(NC(c2cnc(N(C)C)s2)=O)CC1 c1(OC)ccc(C(=O)NCC(C)(O)CNC(=O)C(CC2CCC2)OC)cn1 c1(C(=O)NC(C)CCN(C(=O)C(F)=C2CCC2)C)cc(F)c(F)c(F)c1F C(C)(CC(C)(C)CO)NC(C(C)N(C(=O)CC1C(C)(C)C1(C)C)CCC)=O Cc1nccc(C(N2CCOCC2CN(C(=O)CSc2cn[nH]c2)C)=O)c1O CCCCC(C)C(=O)NCc1nocc1C(=O)NC1CC1CN(C)C C1(C(=O)NC(C(=O)OC)C2CCC2)CC2(CCN(C(C3CNC(=O)N3)=O)C2)C1 c1(OCCC(=O)N(CC(C)NC(C2CC2(C)C)=O)C)cc(F)ccc1F c1(C(N(CC(C)N(C(C2CN(CCC)C(=O)C2)=O)C)C)=O)cnc2n1CCOC2 c1(CNC(C(N)=O)=O)cc(C(=O)Nc2cncc(Br)c2)ccn1 C1(NC(C(=O)NC(C)C)=O)CC2CC(NC(C3(NCC(F)(F)F)CC3)=O)CC12 C1(C(C)NCCCOCCOC)CCN(c2nccs2)CC1 Cc1cccc([N+](=O)[O-])c1C(=O)NC1CCCN(C(=O)C#CC2CCCCO2)C1 C1(CC)CN(C(C)C)CCN1C(=O)NC(c1cn[nH]c1)C CC(C)CC(C)CC(=O)N1CCC(NC(c2cc(O)nc(N(C)C)n2)=O)CC1 C1(C(=O)NC)CCN(c2nnc(C(F)F)n2CC(CC(C)C)OC)CC1 C(C)(CCCNC(C1(C)CC1C(N1CCCC1)=O)=O)NC(CCNC(=O)NC)=O C(C(=O)N(C)C)(C1=NOC2CC12)N1CCC(NCc2cc(C)ns2)C1 c1(C(=O)NC2CCC(CNC(C3(n4cccn4)CC3)=O)C2)ccn2ccnc2c1 C1(CNC(c2ccc(CCC)s2)=O)CCCCC1NC(c1cnc(C)nc1)=O C1(CNC(C2N(C(CNC(=O)OCC=C)=O)CC2)=O)CC1[N+](=O)[O-] c1(C(=O)NC(C2CC(F)CN2CC(N)=O)C)ccc(C(F)F)cc1 C=CC(CC)C(=O)N(C)Cc1cccc(C(C)(C)C)c1 N1(C(C(C)C2CCC2)=O)CCC(C)(C)C(C(=O)NCc2cn[nH]c2)C1 c1(CC)nn(C)c(C(=O)NCC(CCOC)NC(=O)CCC(C)(F)F)c1Cl c1(C(=O)NC(c2ccco2)C)cnn(CCO)c1.C12CC(C1)N2 c1(CC(=O)NCCC(C)(C)NC(C2C(C#C)C2)=O)coc2cc(CC)ccc12 CC1CCCC1(C)NC(c1c(CNC(c2cc(Cl)cn2C)=O)nnn1C)=O N1(C(CC2CC(=C)C2)=O)CCN(C(c2cnn(-c3ccccc3)n2)=O)CCC1C C1(NC(CC2C(C)CCO2)=O)CCC(C)N(C(c2cc(F)ccc2O)=O)C1 CCCC(CC)CCC(=O)N1CCC=C(CNC(c2coc(SC)c2)=O)C1 n1(CC#C)ccnc1-c1nccn1C(C)C(=O)N(C(C)CO)C C1(SC)CCCCC1N=c1[nH]c(N(C)CCF)nc2cc[nH]c12 N1(C(c2nc(OC)oc2)=O)CC(C)(C)OCC1CNC(=O)CCSCC(N)=O c1(C(N2CCC(CN(C(C(n3c(C)ncc3)C)=O)C)C2)=O)cc(F)c(N)cc1F C1(NS(=O)(=O)c2cccc(Br)c2)CS(=O)(=O)C12CCCCC2 c1(C(C)C)ccc(C(=O)NCC2CC(F)CN2C(=O)CCCCO)nc1 CCC(C)(F)C(=O)N1CC(n2cc(CNC(C3CC(=O)N(C4CC4)C3)=O)nn2)C1 C1(C(=O)NC(c2ccc(C)cc2)C(=O)OCC)Cc2ccc(F)cc2C1 C1(C(N(C)CCOCCC(=O)NCC(C)(C)C#N)=O)CCCCC(=O)N1 N#CC12CN(C(=O)Nc3ccc(Cl)cc3)CC1CS(=O)(=O)C2 C1(CNC(=O)NC(C(=O)OC)(C)C)CCCCC1O N1(C(C(C(COC)C)C)=O)Cc2ccc(CNC(=O)CSCCN(C)C)cc2C1 C=CCC(F)(F)C(=O)NCC(C)CN(C(=O)C(C)(O)CSc1cccc(F)c1)C N1(C(C)=O)CCCC1CC(N1CC(C)(C(N2CC(n3cc(C)cn3)C2)=O)C1)=O Cc1cscc1C(=O)NCC1CCN1C(=O)C(C1CCCCC1)O Cn1cnc2c(NC3CCCC3C(=O)Nc3ncc(Br)cc3Cl)ncnc12 Cc1ccc(C(N2CC(C(=O)NCC3(C#N)CCC3)C(F)C2)=O)c(F)c1 C1(C(N2C(C(=O)OC)CC2)=O)N(C(=O)CC2CCC(=O)NC2)CC12CCCC2 Cc1cc(CC(=O)N(C(C(=O)N(C2CCCC2C)C)C2CC2)C)no1 c1(CC(c2ccccc2)NC(=O)NCC2C(C(C)C)CCO2)ccccc1Cl c1(-c2cccc(C(=O)OCC)n2)cc2n[nH]cc2cc1C n1(CC)ccc(CC(=O)NC2C(C(=O)N(CC(O)C3CC3)C)C2(C)C)n1 CC(CC(=O)OCC(C(F)F)n1cccn1)n1cccn1 C1(N(C(c2cnn(C(C)C)c2)=O)CC)CCN(C(C2CC(C)(C)CO2)=O)CC1 Cc1c(C(=O)N(C)CC2COC(=O)O2)sc2[nH]cnc(=S)c12 N1(C(=O)CN2CC3CC3C2)CCC2(NC(C34CC(CC(F)F)(C3)C4)=O)CCCC12 C=CCCCCCCCCCNc1ccc(N2CCN(C)CC2)c(Cl)c1 C1(O)(C(C)NC(C2=C(C)CC2)=O)CCN(C(c2cccc(N)n2)=O)CC1 C1(C2(O)CN(C(C3CCc4ccnn4C3)=O)C2)(CNC(CC(C(C)C)O)=O)CC1 C1(C2CCOCC2)(C(=O)NC2(C)CC(NC(c3ccns3)=O)C2)CC1(F)F CCCC(CC)C(=O)NCCC(C)(C)CNC(=O)COCC=Cc1ccccc1 N12CCCC(CC(C)C)(C1)C2=O.C1(C(=O)N(CCC(=O)OC)CC)CC2CCC1C2 C(=O)(C(CC)C(=O)NCC(C)C(=O)NCCc1cocn1)OCC CP(C)(=O)C(O)C(=O)NCC1COCC1NC(=O)CC1CCC2(CC1)CC2 C12(CNC(C(C3(O)CCC3)NC(C=C(C)C)=O)=O)CC(C)(CCO1)C2 C1(C(=O)NCc2ccc(CNC(C(CC)OC)=O)c(F)c2)CN2CCN1C(C)C2 CCC(CC)(CN=C(NC1CCCC1)N1CC(F)(F)C(F)(F)C1)c1ccccc1 c1(CNC(c2ncccc2F)CC)cc(F)cc(I)c1 C1(C(=O)NCC2(NC(COc3ccc(C)cc3C)=O)CC2)CCn2nnnc2C1 C1(NC(c2c(C)nc(-n3cccc3)s2)=O)CN(C(=O)Cc2cnoc2)CCC1C CC1=CCSC1C(=O)N(CC(O)C(=O)O)C1CCC1 C1(CC=C)(NC(c2ccnc(Cl)c2)=O)CCCN(C(=O)C2=C(C)OCC2)C1 N1(C(=O)COC(F)F)CC2CC1CN2C(C1CCN(S(=O)(=O)C(F)(F)F)C1)=O S(=O)(=O)(c1cccnc1N1CCCC(C)(C)C1)NCC(C)(C)OC N1(C(c2nc(=NC)[nH]c(C)c2)=O)CCC2(CCCN(C(C34CCC3C4)=O)C2)C1 Cc1ccc(F)cc1CNC(=NCCc1cncnc1)NC1CC1C c1(C(=O)Nc2cncc(-c3ccc(-c4ccccc4)s3)c2)cnc2ccccn12 c1(OC(CC)CN(C(C2CCOC2(C)C)C(=O)NCCC#N)C)cccc(Cl)c1 O=C(C1=CCN(C(=O)C=Cc2ccc[nH]2)CC1)NC(CO)CCO CC(CC(=O)NC1CC(C(F)F)C1)C(C)(C)NC(=O)CC(C)(C)C(F)F C1(C(=O)NCC(C)(C)OC(C)C)CCN(C(=O)CN2CCC(C)C2)C12CC2 c1(N(c2c(OCC)cccc2)S(C)(=O)=O)nc2c(C)cccc2s1 N1(C(C2CCC(=O)C2)=O)CCN(C(c2cc([N+](=O)[O-])n[nH]2)=O)CC1CC1CC1 N1(CC(=O)NC2CCC(NC(C(C=C=C)C)=O)CC2)CCP(C)(=O)CC1 CCCCC(C)CCC(=O)NCC(c1ccccc1F)NC(c1sncc1C)=O C=C(C)C1CN(C(C2(C)C=CCN2C(c2ccc([N+](=O)[O-])[nH]2)=O)=O)CCO1 Cc1nn(CC(=O)NCC(C)(C)C(=O)NCCCCCF)c(=O)o1 C1(NC(C2(COC)C=CCN2C(=O)C=CC2CCC2)=O)CCCCC1(C)C C1(NC(c2c(CC)n(C)nc2)=O)CN(C(c2nccn2C(C)C)=O)CCC1CO CC1=C(C(=O)N2CC(CC(=O)NCC(Cl)C(C)(F)F)CC2(C)C)CCCO1 C1(CNC(=O)C(O)C2CCCC2)CC2(CO1)CN(C(C1(C3CC3)CCCO1)=O)C2 N=c1ccc(C(N2CCC(OC3CC3)C2)=O)c(Cl)[nH]1 c1(CC(=O)NC2C(NC(CC=CC)=O)COCC2)cc(C)cc(F)c1 N1(C(CC(CC)CC)=O)CC(C)CN(C(c2coc(Br)n2)=O)C(C)C1 c1(OC)nc(Cl)ccc1C(=O)N(C(C)CCNC(=O)CC(=O)N(C)C)C C(C(C)(C)C(=O)N1CC(O)CC1C(=O)NCCC1CCCCO1)OCC C1(C(C)C)N(C(c2cscn2)=O)CC12CCN(C(=O)CCC1CCC(C)O1)CC2 c1(C(N2CCC(CN(C(c3cc(OC)n[nH]3)=O)C)C2)=O)cncc(F)c1Cl N1(C(CCC(C)O)=O)CC2CCC1CN2C(c1coc(C2CC2)n1)=O CCCC(C#N)C(=O)NCCCCNC(c1cc(C)ccc1NS(C)(=O)=O)=O C(=O)(CC(C)C(F)(F)F)NC1(CCC(=O)Nc2cccc(OC)c2O)CCCC1 C1(NC(=O)CC2(O)CCC2)CC2CC1N(C(c1ccc(F)s1)=O)C2 C1(C(CC)=O)CCC(C(=O)NN2CCC2Cn2cc(CCC3CC3)nn2)CC1 Cc1cc(CNC(=O)C(C2CCC2)NC(c2cccnc2C)=O)cc(C)n1 C(CC)(C(=O)NCCC(C)(C)NC(C1CCCC1C)=O)=CC N1(C(c2n(CC)ncn2)=O)CC(NC(=O)CCC(=O)c2ccc[nH]2)CC1(C)CC C1(C(=O)NC2(CNC(CCC(=O)NCCC)=O)CCCC2)CNC(=O)CC1C N1(C(C(C)(C)O)=O)CCC(C(=O)NC2CCN3CCC2C3)C(O)C1 C1(N(C(CSCCC)=O)C)CN(C(c2cc(C(=O)OC)sc2C)=O)CC1O O=C1CNc2ncc(C(N3CCC(c4cncc(F)c4)C3)=O)cc2N1 C(=O)(CC1OCc2ncccc21)NCC1CC(C)(C)CN1C(=O)C(F)C(F)(F)F N1(C(c2cc(C)c(O)nn2)=O)CCC(C)(C)C(C(N2CC3CC2(CO)C3)=O)C1 CC(N)(CS(C)(=O)=O)C(=O)NCc1nc2cc(F)ccc2s1 c1(C(=O)NC(COC)C2(C)CC2)c(-c2ccccc2)coc1C C1(C(=O)NCCC2CCCN(C(C3CC(SC)C3)=O)C2)(CC)CCCCO1 c1(OC)ccc(C)c(C(=O)NCC2CCC(C)CN2C(c2cscc2F)=O)c1N C1(NC(C2C(C)C2)=O)CC2CCC(C1C)N2C(=O)CCC1CC(C)(C)CO1 N1(C(CN(C(C)C)C)=O)CC2(CCC(NCc3cc(F)cc(Br)c3)C2)C1 CC(C)CC(C)C(=O)NC1(CC=CC(=O)NC(C)Cc2cn[nH]c2)CCC1 c1(C(=O)NC2CC(NC(c3c(CC)cccc3CC)=O)C2)cc(S(N)(=O)=O)c[nH]1 CC1CN(C(=O)CNS(=O)(=O)C2CC2)CCC1CNC(=O)Cc1ccccc1F N(C(=NCCc1ccc(F)cc1)NCCCS(=O)(=O)N(C)C)C1C(C)CSC1 C(=O)(CC(CN(C)C)CC)N1CC(C#C)(C(=O)NCC(O)CCC)C1 C1(N=[N+]=[N-])(C(=O)NC(C)CCNC(=O)CCCC2CCCO2)CCOCC1 N1(C(c2c(F)ncc(C)c2)=O)CCCC2CN(C(c3c[nH]cc3C)=O)CCC12 C(C(N=[N+]=[N-])C(=O)NCCCOCCC(=O)N(C1COCC1O)C)OC c1(C(N2CCC(C(=O)NCCCCN(C(C)C)C)C2C)=O)ccc2cc[nH]c2n1 c1(CC)nocc1C(=O)NCC1C=CCN1C(C1CC1C(C)C)=O c1(CC(N2C(CNC(Cc3nnc(C)s3)=O)CC2)=O)csc2ccccc12 C(CC(C)C(=O)NC1(c2ccccc2)CN(C(=O)C(OC)OC)C1)=CC N1(C(CCC2CCC(=O)C2)=O)CCOC(CCCNC(=O)CC2(C(F)F)CC2)C1 c1(CC(c2n(C(CC)C)nnn2)NC2CN(c3cnccn3)C2)cccc(Br)c1 Cc1cc(Cl)cc(NC(C2CC(F)CN2C(c2ccc(Cl)s2)=O)=O)c1Cl CCC(F)(F)CC(=O)NCC1(F)CCC(NC(c2cccc(CF)c2)=O)C1 N1(C(c2c[nH]c(=NC)s2)=O)CC2(CCN(C(C3CCCN3C(=O)NC)=O)C2)C1 C1(C(N2C(CCOC)CN(C(=O)CCC(C)(C)O)CC2)=O)CCCCC12CCC2 Cc1ncc(C(=O)NCCC2CC(NC(C3(n4cccn4)CC3)=O)C2)n1C CCC(C)(CCC(C)C)C(=O)N(CCCCNC(c1c[nH]cc1Br)=O)C C1(C(=O)NCCN(CCC)C(C2CC3(CC3)C2)=O)(COC)CCCCO1 C(CCC(O)C(=O)NC(c1cn(C)nn1)C)NC(C=C(C)C)=O C1(NC(c2[nH]cc(OCC)c(=O)c2)=O)CC2CC(C1)N(c1nc(C#N)c(Cl)s1)C2 Cc1c(C(N2CCC(C(C)NC(c3snc(Cl)c3Cl)=O)C2)=O)ccn1C1CC1 c1(NC(C23CC(NC(C(CC(C)C)O)=O)(C2)C3)=O)cccc(Cl)c1C#N Cc1nc(O)[nH]c1C(=O)NC1CCC(CCNC(C2(C)CC2(C)C)=O)C1 c1(C(N2CC(NC(CC(C)F)=O)CC2(C)C)=O)ccnc2ccc(F)cc12 N1(C(CCCC(=O)NCC)=O)C(CNC(=O)C(O)C(C)CC)CC2COCC12 CCCCC(C)CCC(=O)N1CCC(NC(c2cc(C#N)ccn2)=O)C1 C1(C(=O)NC2C3CN(C(=O)C(C4CCCCC4)O)CC23)CCc2ncncc2C1 c1(C(=O)Nc2c(C)ccc(C(=O)N(C)C)c2)cc(S(=O)(=O)NCC(C)O)c[nH]1 c1(OCC)oc(C)nc1C(=O)NC1C2CN(C(=O)C(C)(O)c3ccccc3)CC12 CON1CCC(C(=O)N(C2(C(=O)NCc3cncc(O)c3)CC2)C)CC1 C(=O)(CC(CC)C(F)F)N1CCCC(N(C(CCC#CC)=O)C)CC1 CCCCCC(O)C(=O)N1CCCC(C)(NC(C2CCC(C3CC3)CC2)=O)C1 c1(OC)cnc(C(=O)NC2(CCO)CN(C(=O)C=C(C)C)C2)c(F)c1 N1(C(C(C)OCC)=O)C2CCCC1CN(C(=O)CC1CCN(CC(F)F)CC1)C2 N1(C(CCCOC)=O)CCC(C)(NC(=O)Cc2ccsc2Br)CC1 N1(C(C(CCOC)C)=O)CC2(CCC(CNC(=O)CCC(=O)N(C)C)O2)C1 c1(OCC)nc2ccc(C(N3CCN(C(=O)CSC)C(C)C3C)=O)cc2[nH]1 C(CCC(C)(C)C)(C(=O)O)NC(CC(CC)(C)C)=O c1(CCC(=O)NC2CC(C)(NC(CCC=C)=O)C2)ccccc1C(N)=O Cc1cc(C(N2CCCCC2C(=O)Nc2cccc(Cl)c2Cl)=O)ccc1C#N c1(C(N(C2CC(c3nncn3C)C2)C)=O)cc([N+](=O)[O-])n[nH]1 c1(C(=O)Nc2c(C(N)=O)ncc(Cl)c2)ccc2ncc(C3=CCCC3)n2c1 Cc1ccc(NC(C2CCN(C(=O)C(O)C(F)(F)F)CC2C)=O)cc1O C1(C(=O)NCC2N(C(c3cncc(C)c3)=O)CCOC2)CN2CCC1CC2 C1(C(=O)NC(CNC(CS(=O)(=O)NCC)=O)C2CC2)CC2(CCC2)CO1 c1(SC(C(N2C(C(=O)OC)CC(O)C2)=O)C)cc(-c2ccccc2)sc1SC n1(CC(N2CC3C(CNC(C4CC(SC)C4)=O)(C3)C2)=O)cnc([N+](=O)[O-])c1 c1(Cn2cc(C(N(CC(C)N(C(CCSC)=O)C)C)=O)nn2)cccc(Cl)c1 N1(C(C2(CF)COC2)=O)CCCOC(CNC(C2(CO)CCCO2)=O)C1 C1(C(N(OC)Cc2cccnc2)=O)CCCN(C2CCCCC2C(=O)N)CC1.OC c1(C(N2CC(NC(c3n(C)ccn3)=O)C3C2C3)=O)cc2c(cn1)OCCC2 Cn1nc(CNC(=O)CCN(C(=O)COc2ccsn2)C2CC2)oc1=O CCC(C(=O)NCC1CCC(F)(CNC(=O)CCn2ccc(C)n2)C1)C(C)C C(=O)(CCCC(=O)NC1CCCCC1CNC(=O)CNC(C1CCC1)=O)NCC N1(C(C(C)N(C(C)=O)C)=O)CCCCC1CCNC(c1cnco1)=O CC1CN(C(=O)CCCC#N)CCN1C(=O)Cc1ccon1 C1(NC(c2ncn(C(C)C)n2)=O)CN(C(=O)CC#N)CC1C C(=O)(C(C)CC(=O)OC)NC(CCOC)CNC(c1ncc(F)cn1)=O C1(C(=O)NCC2CN(C(c3[nH]cc(CC)c3)=O)C2)NC(=O)CC1C(F)(F)F N1(C(C(=O)Nc2ccc(OCCC)cc2)=O)CCC12CCS(=O)(=O)C2 C12(COCC)CC(C1)C(NC(C1(NC(C3CCCO3)=O)CCCC1)=O)CO2 Nc1cc(C(=O)NCC(C2CC2)NC(=O)CCC2CCCO2)c2ccccc2c1 Cn1cc([N+](=O)[O-])c(CC(N2CCN(C(=O)COC3CCOC3)C(CF)C2)=O)n1 C1(C(=O)NCC2(COC)CN(C(C3CC(F)(CF)C3)=O)C2)CCNC(=O)C1 C1(NC(C2ON=C(C)C2)=O)CCN(C(c2ccc(Br)cc2C)=O)CC1F C1(c2nnnn2-c2ccccc2OC)(NCC(CC)(C)C)CCCC1OC Cc1cc(C(=O)NCC2CC2CNC(C2(C)CCCC2(F)F)=O)c(C)cc1Cl n1(CC)cc([N+](=O)[O-])c(C(=O)NCC2CCC(CN(C)C(C3CC3F)=O)CC2)n1 C1(NC(CC(=C)C)=O)C2CCCN(C(=O)CC3CCCCN3C)C2C1(C)C C(C)(c1ccco1)=CC(=O)NCCOCC(N1C(C)(CCC)CC1)=O Cc1nc(C=CC(=O)NCCN2CCC(NC(C3CC(Cl)(Cl)C3)=O)CC2)cs1 N1(C(c2cn(C)c(Br)c2)=O)CCC(NC(=O)C=CCN2CCCC2)C12CC2 CCC(C#N)(CC)C(=O)NCC1CN(C(=O)Cc2ccc(Cl)c(Cl)c2)CCCO1 C1(=CC(=O)NCCN(C(=O)C(C2CCOC2)OC)CC)CCC(C)(C)CC1 N1(C(c2nc(CC)sc2)C(=O)Nc2c(C)csc2Cl)CCCN(C2CC2)CC1 N1(C(CC2CCC(C)CC2)=O)CC2CCCC(CNC(c3cscn3)=O)C2C1 N1(C(C)C)C(=O)CCC1C(=O)N(C1CCN(C(c2ccc(C(N)=O)nc2)=O)C1)C Cc1ccncc1C1CCN(C(=O)NCc2ccoc2C(F)(F)F)C1 C1(C(=O)NC(C2CCCC2)CNC(C2CCC(COC)O2)=O)CC2CCC1CC2 CC(C)C(O)C(C)C(=O)NC(CC1CCC1)C(=O)NC1CC2(C1)CC(C)(C)C2 C1(NC(CC2OCCN(C(CCc3ccn(C)n3)=O)C2)=O)CCC2(CCC2)CC1 c1(C(=O)NCCC(C)NC(C(CN(CC)CC)F)=O)ncnc(OC(F)(F)F)n1 c1(N(C2CN(C(C(C)(C)C)=O)C2)C(Cn2ncc(C#C)c2)=O)ccc2ccn(C)c2c1 C(=O)(C1=CCC(F)(F)CC1)NC1(C)CC(NC(c2c(C)nc(C)s2)=O)C1 c1(C2(CNC(CC(c3ccccc3)SC)=O)CC2)ccc(C(N)=O)cc1 Cc1cc(CCC(N2CC3C(C2)C3(C)C)=O)cc(C)n1 c1(C(N(C(C)CNC(=O)CP(C)(C)=O)C)=O)cc2c(o1)CCCC2 CC#CCCCC(=O)NC1CCCCC1n1cc(CC2CCCOC2)nn1 c1(C(N(CC(C)C(=O)N(CCC(F)(F)F)C)C)=O)cccnc1S N1(C(c2c(O)ncc(CC)c2)=O)CC(C)CN(C(=O)CCCOC(C)C)C(C)C1 CC1(CC(=O)NCCCN(C(c2ccn(CC(F)(F)F)n2)=O)C2CC2)CCCO1 C(c1cnccn1)=CC(=O)N(C1CCN(C(C2CC(C#N)C2)=O)CC1)CC Cc1cnc(CCC(=O)N(C(C)CNC(=O)Cc2cncnc2)C)[nH]1 C1(CSC)CCN(C(=NCCc2c(C)nn(C)c2C)NCc2cc(C)on2)C1 C1(NC(COCc2onc(C)n2)=O)CC2CCC(C1)N2C(=O)CC1(O)CCCOC1 C=CC(CC)CC(=O)N(CC(=O)NCCc1noc(=O)n1C)CC=C N1(C(CC(CC)OC)=O)CC2(C(=O)NC3C(O)CC3O)CC1CO2 CC1CCC(NC(c2ccccc2OCC2CC2)=O)CN1C(=O)CCCCF C1(NC(C=C(C)C)=O)CCN(C(=O)CCC(=O)c2cccc(N)c2)CC1F c1(C(=O)NC2CC(F)(CNC(c3cnco3)=O)C2)csc2ncnc(O)c12 N1(C(C2N(CCC)CCC2)=O)CCC(C)N(C(c2nnc(S)n2C)=O)CC1 Cc1cc(C(=O)NC2CC3(C2)CC3NC(=O)C=Cc2cncc(O)c2)cc(O)n1 C1(OC)CCN(C(C2(NC(=O)CCCN(C)C)CCN(C)C2)=O)C(C)C1 C=CC(C)(O)CC(=O)N1CC(NC(=O)Cc2cnsc2)C(n2ccnn2)C1 c1(C(N(CCCNC(=O)C(C)(C)CF)CC)=O)cc2c(Br)cccc2cn1 N1(C(C(c2ccn(C)n2)C)=O)CC(NC(=O)CN2CCC(O)CC2)C2CCCC12 N1(C(N2CC(C(=O)NC(CC)C(=O)c3ccccc3)C2)=O)CCCCC1C(C)C C1(C(=O)NC(C2CCN(c3ncnc4[nH]ccc34)C2)C)CC(C)(C)CC(C)(C)C1 C1(NC(c2nc(C)[nH]n2)=O)CC=CCC1C(=O)NCCC(C)C c1(CNC(c2n(CC)nnn2)c2cc(C(N)=O)cs2)c(F)cccc1I N1(C(c2nc(OCC)oc2)=O)CC(CNC(=O)CC23COCC(C2)C3)CC1(C)C c1(CC(N2CCC(O)(CN(C(C(C=C)O)=O)C)CC2)=O)ccc2sccc2c1 c1(C(=O)NCC2(OC)CN(C(=O)CC3CCC(=O)N3)C2)cc2c(O)cccc2[nH]1 C1(N(C)C)CCCC(C(N2CC(N3CCN(C(C4C5CCCC45)=O)CC3)C2)=O)C1 c1(C(=O)NCCN2CCN(C(CC#C)=O)CC2=O)ccc(F)c(C(F)(F)F)c1Cl Cc1c(F)cc(CNN2CCN(C(c3cccc(O)c3C)=O)CC2)cc1F Cc1ccc(CCNC(=O)CCCc2cnccn2)cc1F C(=O)(C(CC(C)C)ONC(C1CC(=O)C1(C)C)=O)N(c1ccccc1)CC Cn1cnc2c(NC3CCCC3C3CC3)[nH]c(=NCC34CCCN3CCC4)nc12 C(=O)(C1c2ccccc2CN1C(=O)C(C)(O)C(F)(F)F)Nc1c(OC)nn(C)c1 c1(CC)nc(N2CC(N(C)C(c3cccc(C(=O)OC)n3)=O)C2)cc(C)n1 C12(OC)CCC(C(=O)N(CCCNC(=O)C(F)OC(F)(F)F)C(C)C)(CC1)C2 N1(C(C(CC)(C)CO)=O)CC2(C=C(C(=O)NCCC(C)F)CO2)C1 c1(C(=O)NCC23CCC2CN(C(=O)CC2CC2(Cl)Cl)C3)ccc2[nH]ccc2c1 C1(=O)C(C)(OCC(=O)NC(C)CCCc2n(CC)ncc2)COC2CN1C2.OC.OC c1(C(N2CCCC(O)(CNC(c3cnon3)=O)C2)=O)ccc(Br)c(F)c1F N(C(=NCCC(C)=O)NC1CCC(C(N)=O)C1)C1CCN(C(=O)OCC)CC1 C1(C(=O)NC(C=C)C)(CCNC(=O)Cc2nonc2C)CCCC1 C(=O)(C(CC1CCCC1)NC(=O)C(O)CN(C)C)N(CC(C1CC1)OC)C C1(C(N2CC=CC(NC(c3n(CC)ncn3)=O)C2)=O)CC2CC2CC1C C#CC1CN(C(C2CN(C(=O)COCCCF)CCO2)=O)CCO1 N1(C(c2ccc(OC)nn2)C(=O)NCCC)CCN(CCOC)C(=O)C1 C(C1CN(C(c2ccccc2I)=O)Cc2ccccc21)NC(=O)C1CC1 c1(C(=O)NCCCCC(C)NC(c2cc(C(N)=O)n(C)n2)=O)ncc(Cl)cc1Cl C(CN=C(NCC(O)CN1CCOC(C)C1)N1CCC(O)(CC)CC1)OCC C1(C(=O)NC(CC(C)NC(c2c(C)nn[nH]2)=O)C)CCCCC(=O)C1 C(CC(C)C(=O)NCC(C)CN(C)C(c1cc(C(F)F)nn1C)=O)=CCC C1(C(=O)NC2CC(C)C2)CN(C(c2ccc(Br)cc2)=O)CC1C C(=O)(C(C)(C)C(F)(F)CC)N1CCC(N(C(c2noc3c2CCCC3)=O)CC)C1 c1(NC=O)ccc(C(=O)NC2CCC(F)(CNC(C3CC4CC4C3)=O)C2)cc1 c1(NC2C(C)Cc3ccccc32)[nH]c(=NCc2ccc(C#N)o2)nc2sccc12 c1(CC(N2CCC(O)(CNC(CCS(=O)(=O)NC)=O)C2)=O)cc(F)cc(C#N)c1 N1(C(C(=O)NCC)C2CC2(C)C)CC(C)(C)C1OC(CCC(=O)OC)=O c1(-c2nnc(C(C)ON3CCC(CC(N)=O)C3)o2)ccc(Cl)c(Cl)c1 C12(CNC(c3cc(C)oc3)=O)CN(C(c3cnc4ccsc4c3)=O)CC1CCO2 c1(CC(N2C(C(=O)Nc3ccc(SC)cc3)CC2)=O)cc(F)ccc1F N1CC(O)C(O)C1.C(C(O)CC(C)CCCC)n1cc(COCCOCC)nn1 c1(CC(=O)NCC(CC)NC(C2CCCC(C(C)(C)C)C2)=O)nnc(S)n1C c1(C(N2CCC(N(C(C3C(C)C3)=O)C)C2)=O)nc2ncc(Br)cc2[nH]1 c1(SC)nc(C(=O)NCCCNC(C23CCCN2CC(O)C3)=O)c2ccccn12 Cc1ccc(F)c(C(=O)NCC(C)(CO)NC(c2ccc(C3CC3)nc2)=O)c1 c1(-c2scc(NC(C3CCC(O)CC3)=O)n2)c(Cl)cccc1Cl Cc1cc(C(N2CC=C(C(=O)NCCCCCO)C2)=O)nnc1C C1(NC(C2CC(C)OCC2)=O)CC2CC1CN(C(c1ccsc1C(F)(F)F)=O)C2 CCC(O)C(F)(F)C(=O)N(CC(CC)NC(=O)Cc1ccc(F)c(OC)c1)C c1(OC)ccc(O)cc1C(=O)NC(C)(CNC(c1ccc(C(C)F)cc1)=O)CO c1(CC(=O)NCC(CN(C(COCCCC#C)=O)C)C)ccc(Cl)cc1F CCN=c1[nH]cc(C(=O)NCC2CN(C(=O)C(O)P(C)(C)=O)C(C)(C)C2)s1 c1(C(=O)NC(C2CC(NC(C3CC(CC4CCC4)C3)=O)C2)C)cnc(C(F)F)s1 C(C(CNC(=O)Cc1cnc[nH]1)C(F)(F)F)NC(=O)CN1CCSCC1 c1(NC(C(=O)NC(C(C)NC(CC=C)=O)CO)=O)nc(C(C)C)c(C)s1 C1(COC)CCCN(C(c2ccn(CCNC(c3cc(C)nn3C)=O)c2)=O)CC1 C=CCC(CC)C(=O)N1CCCC1C(C)NC(c1ncc(C)cn1)=O C1(NC(Cc2cc(C)on2)=O)CCCCC1NC(C1CCCCS1)=O N1(C(=O)Nc2nnc(-c3ccc(F)cc3)s2)CC2CC(C1)C2(F)F C=CC(CCC)CC(=O)N1CC(O)(CNC(c2cc(C3CC3)ncn2)=O)C1 Cn1nc(Br)nc1CNC(c1nnnn1C(C)(C)C)C1(c2cccs2)CC1 c1(C(=O)NCC(CC)NC(=O)CN2CCC(CO)CC2)c(C)nn(CC)c1Cl c1(C(=O)NCC2C(NC(C(C)NC(C)=O)=O)CCC2)cccc2c1OCCCO2 c1(C(N(C2CCN(C(=O)C(C3CCCC3)SC)C2)CCC)=O)coc(C2CC2)n1 Cn1nc(C(N2CC3CN(C(=O)Cc4ccsc4)CCC23)=O)c2c1CCSC2 Cc1cccc(C(N2CCC(CF)(NC(=O)CC3CCC(=O)NC3)C2)=O)c1O N1(C(C(CCCC)O)=O)CCC2(CC1)CC2NC(C1(F)CCCCCC1)=O C1(C)(C(=O)NC(C)CCN(C)C(C2CCC(C)O2)=O)CCS(=O)(=O)CC1 Cc1cc(C(N2CCN(c3ccnc(-c4ccccc4)n3)C(C)C2)=O)nc(C)c1 CC1CC(C)(C(=O)Nc2cnc(Cl)c(CNc3cnc(F)cn3)c2)CCO1 Cc1cc(C)c(C(=O)NC2CC2CNC(c2cc(C#N)c[nH]2)=O)c(O)c1 Cc1cccc(C(=O)NC(C)C(=O)NC23CC(C2)N(C(C2(O)CCC2)=O)C3)c1 N1(C(c2c(CC)nns2)=O)CCC2(CC1)CC2NC(=O)C(CC)SC CCC(C)CCC(=O)N(C1CCN(C(=O)CCOC2CCCCC2)C1)C N1(C(Cn2cnc(C)n2)=O)CC(C)(C)C(O)C1(C)C C1(C(N2CC(O)(C(C(N3C(CC(N)=O)CCCC3)=O)F)C2)=O)CCOCC1(C)C c1(CN2C(C(=O)NCC3(N(C)C)CCOCC3)COCC2)c(Br)cc(F)cc1Br c1(C(N(C=O)CC2CCC2C(F)(F)F)C)nncn1Cc1ccccc1 C(=O)(C(C(C)C)N(C)C)NCC(C)(C1CC1)NC(C(c1ccccc1)SC)=O c1(OC)ccc(Cl)cc1-n1nc(C(C)C)nc1C1COC(=O)O1 C(CC)(C(=O)NC1(C(=O)NC(C)(C)CCN(C)C)CC1(C)C)OCC C1(C)(C(N2CCN(C(C3=CC(C)(CC)C3)=O)C(CO)C2)=O)CCS(=O)(=O)CC1 C1(C2CC2)(CNC(c2nc(CC)sc2)=O)CCN(C(c2cc(O)cc(Cl)c2)=O)C1 C(=O)(C1CCc2c(Cl)cccc21)NC1CC(N(C)C(c2cn[nH]c2)=O)C1 N1(C(C)C)CCN(CCC(=O)NCC(O)CN(C)C(C2CCCS2)=O)CC1 O=C1OC2CON(C(=O)c3cc(-c4ccncc4)[nH]n3)CC2O1 c1(C(=O)NCCN2CCN(C(C3(O)CCC(CC)C3)=O)CC2)cc(F)ccc1O CC(C)CC(C(=O)N1CCN(C(C2CCC(N(C)C)C2)=O)C2(CC2)C1)C(C)C S(=O)(=O)(c1cn(C(C)C)cn1)N1CCC(C=C)(C(=O)O)C1 c1(NCCCN(C2CCCC(O)C2)C)ccc(Cl)cc1 C1(CN(C)C(C2CC23CC3)=O)CCN(C(c2csc(Br)c2)=O)C1 C1(CNC(CCNC(C)=O)=O)CC2CCC1N2C(C1(C)CC2CCC1C2)=O CC(CC(=O)N(CCCN(C(=O)C=C1CCSCC1)C)C)C1CCCO1 c1(OC)cccc(-c2nc(C(C)COC)n(C(C)C3CC3)n2)c1 C1(NC(=O)CSc2ccccn2)CC2(NC(=O)CSn3cnnn3)COC1C2 C(C)(C)(CCC(=O)N1CCCC(CO)(Cc2cn(CCN(C)C)nn2)C1)OC c1(CC)ocnc1C(N1CC(CF)(NC(c2csc(=N)[nH]2)=O)C1)=O C1(NCc2ccc(C)nc2)CC(NC(c2cnc(Cl)s2)=O)C12CCC2 C1(NC(c2c(CC)nn[nH]2)=O)(CNC(C2CCCC(CC)C2)=O)CCCCCC1 c1(CC)ccc(C(=O)NCCC2(O)CN(C(c3cc(Cl)nc(=N)[nH]3)=O)C2)c(O)c1 N#Cc1ccc(=NCC(=O)N2CC3(CCN(C(C4(CF)CCC4)=O)C3)C2)[nH]c1 CCCC(O)CC(=O)N1CC2CC(NC(c3ccccc3OCC3CC3)=O)C2C1 n1(CCC)nc(C)c(C(=O)NCC2(F)CN(C(C34CC(F)C3C4)=O)C2)c1C C(=O)(C1=CC2CCCC12)NCC(C)(C)NC(=O)C1=CCCOC1 c1(C(=O)NCCOCCNC(CCC=C=C)=O)ccc(CC)c(N)c1 C1(CC)CN(C(c2ccccc2Cl)=O)CCC1NC(=O)CSc1cccc(C)c1 n1(CC)nnc(C)c1C(=O)NCC(C)NC(c1cnoc1-c1ccccc1)=O C1(CCC)CN(C(=O)C(C)CC(N)=O)CCN1C(=O)CCc1ccc[nH]1 C(=O)(C(F)(F)C(F)(F)F)N(CCCNC(C(C)(C)NC(=O)OC)=O)N(CCC)C c1(C(=O)NC2CCN(C(C3ON=C(C)C3)=O)C2C)csc2cc(Cl)ccc12 C(=O)(CC(C(C)C)c1ccon1)NCC(=O)OC.c1(O)ccc(NCCCC)cc1 C1(CCOC)CN(C(=O)CC#N)CCN1C(c1cncc(OCC(F)(F)F)c1)=O CCC(CCC(=O)NC(C)(CNC(c1cc(C)cc(C)n1)=O)C1CCC1)OC CCC(C)(CCC(C)C)C(=O)N1CCCC(CNC(=O)CC(C)(C)CSC)CC1 C1(C(=O)NC2CCC2)(COC)CCN(C(C2CC2c2sccc2C)=O)CC1 S(=O)(=O)(c1ccc(C#N)c(NCCc2ncoc2C)c1)N1CCC(CC)C(C)C1 CCC(C)(C)C(=O)NCCC(Cc1ccccc1)NC(=O)COCC1CCOC1 C1(CNC(=O)CCCc2nccs2)CCN(C(=O)CCOC2CCC2)CC1 C=CCC(C(=O)NCC=CCNC(c1occc(=O)c1OC)=O)C(C)C Cc1ccc2c(=NCC3CCC4CC34)[nH]c(=NC3CCN(CCF)C3)[nH]c2c1 C1(C(=O)NCCN(C(CC=CCC)=O)CCCN(C)C)CCCCN1C(C)C C(=O)(CCS(=O)(=O)N1CCOCC1)N(C(C)CN(C)C(C1(C2CCC2)CC1)=O)C c1(C(C(=O)NCCCSC)NCCCN(CC)CC)ccc2ccc(Cl)cc2n1 N1(C(c2c(OC)cncn2)=O)CCC2CCCC12C(N1CCC(F)(CF)CC1)=O CC(C)CC(=O)NC(C(=O)NCC1C2COCC12)C1CCC1 C1(NC(CSCCC(C)C)=O)CC(O)CN(C(c2ccnc(OC(F)F)c2)=O)C1 S(=O)(=O)(c1ccc(NCCc2cn(CC)nn2)c(Cl)c1)N(C)CC1CC(=C)C1 Cc1cc(C(=O)NC(C2CCCN(C(=O)C=CCO)C2)C)cc(O)c1 c1(C(N2CC(N(C)C(c3ncn(C)n3)=O)C(F)C2)=O)cc(Cl)cc([N+](=O)[O-])c1 C1(CNC(C2(C(N)=O)CC2)=O)CCN(C(c2nn[nH]c2Cl)=O)C12CC2 c1(NC(c2c(CC)csc2)=O)cccc2c1OC(C)(C)C2 CC(C)C(O)C(=O)NCC1(C)CC(NC(=O)CSc2cn[nH]c2)C1 Cc1cc(C)c(-c2nc(C3CN(C)CCO3)nn2C(C)C(C)C)[nH]1 Cc1c[nH]c(CC(N)=O)c1C(=O)NC1CCC1NC(c1n[nH]cc1Cl)=O O=C(C(O)C(F)(F)F)NC1CCCCN(C(=O)C(O)Cn2cncn2)C1 n1(CCOC)c(N2CCC(F)(COC(C)(C)C)C2)nnc1-c1sccc1O c1(C(=O)NC(CC=C)CNC(=O)C(C)CSC)nc(-c2cnn(C)c2)oc1C Cc1noc2cc(C(N3CC(CNC(C4C(C)(C)C4(C)C)=O)C4CC34)=O)ccc12 C1(NC(C2CC(O)(CC#C)C2)=O)CN(C(=O)C(c2ccc(F)cc2)F)CCC1C C1(CNC(C(C)NC(=O)NC)=O)CCN(C(c2cnn(CCO)c2)=O)C(C)C1 C(=O)(C(O)C(C)(C)C)N(CCNC(C1(C(=O)OCC)CC1)=O)C CCCC(CC(=O)NCc1ncccc1O)NC(=O)C(O)CC N1(C(C23CC(C)(C2)C3)=O)CCN(C(=O)Cn2nc(C(C)(C)C)cc2N)CC(O)C1 c1(C(=O)NCCCC2N(C(c3c(C)nn[nH]3)=O)CCC2)ccc2nc(O)cn2c1 C(=O)(C1CCOc2ccccc21)NCC1(F)CC(CNC(=O)CO)C1 c1(CC)ccc(C(=O)NCCCn2cc(-c3ccc(C(C)C)cc3)nn2)cn1 N1(C(C2CNC(=O)N2)=O)Cc2nccn2CC(NC(c2cc(F)cc(Cl)c2)=O)C1 N1(C(C(CC)N(C)C)=O)CCC(CNC(c2ccc(-c3ccco3)[nH]2)=O)C12CC2 c1(C(N2CC(F)(C(N3CC(CC#C)OCC3)=O)C2)=O)ncc(N)cc1C c1(C(=O)NC2C(C)N(C(=O)COC3(C)CCCC3)CC2)cc2n(n1)CCCC2O N1(C(C(=Cc2cnc[nH]2)C)=O)CCN(C(c2nc(C)ccc2F)=O)CC1C1CC1 N1(C(C(CC)=CC)=O)CCC2(CC1)CC(NC(=O)Cc1cncn1C)CO2 N1(C(C(C)OCCC=C)=O)CC2(NC(=O)C(O)C3CC3)CC1C2 c1(C(=O)NCC(C)(C)OCCNC(C(F)=C(C)C)=O)ncc2ccccn12 C=CC(CC)CC(=O)C(N1CC(C(=O)ON2CCCCC2)C(O)C1)=O N1(CC(=O)N(C2C(C)CCCC2)C)CCC2(CC1)CN(C(C1(C)CC1)=O)C2 n1(C(C)C)nccc1C(=O)NC1COCC1NC(c1ncn(C(C)(C)C)n1)=O C(=O)(C(C)S(N)(=O)=O)N(C)CC1CCN(C(C=C(CC)CC)=O)C1 CC(C)CC(C(=O)N1C2CCC(C2)C1CNC(C1CC1C)=O)n1ccnc1 C1(C)(N(C2COC(CC(C)C)C2)C(C)=O)CCCN(c2ccccn2)C1 c1(NC(c2nccn2-c2ccccc2)C)nccc(=NC2CCOCC2F)[nH]1 N1(C(C(C)=CC2CC2)=O)CC(C2CCN(C(c3cnc4scc(C)n34)=O)CC2)C1 C(=O)(C1Cc2c(Cl)cccc21)NC(CNC(c1ccc(OC)cc1)=O)(C)CO c1(C(N2CCN(CC3CCCC3)CC2C)C(=O)NCC(C)C)cccn(C)c1=O N1(C(C2CC(n3cc(C4CCN(C)CC4)nn3)C2)=O)CCc2cccc(O)c2C1 N1(C(C2C3(CC(NC(C(C(C)OC)N(C)C)=O)C3)C2)=O)CC(C)CC(O)C1 CCCCC(F)C(=O)NCc1cc(C(=O)NCC2CCCC2O)n(C)n1 CC(C(=O)NC(CNC(=O)CC1CC2(CCO1)CC2)C1CCC1)C(C)(C)C c1(OC)cccc(SCC(N2CC(N(C(=O)CSC(F)F)C)C(O)C2)=O)c1 N1(C(C(COCC)n2cc(Cn3cc(C)cn3)nn2)=O)CCC2(C=CCO2)C1 C1(CNC(c2c[nH]nc2-c2ccncc2)=O)(NC(C2CCC2(F)F)=O)CCOC1 c1(OC)ccc(F)c(C(N2CC(CNC(C3C(C)C3(F)F)=O)CC2(C)C)=O)c1 CCC1=NOC(CC(N2CC(CC(F)C(=O)NC(C)(CC)CC)C2)=O)C1 C(=O)(C1=CCOCC1)NCC1(C(N2CCC(CC(N)=O)C2)=O)CC2(CC2)C1 C1(CNC(CNC(CCC)=O)=O)C(C)CCCN1C(c1cn(C2CC2)cn1)=O c1(C(N(CCCCC)C)=O)occc1CNC(c1ccncc1)=O N1(C(=O)OC(C)(C)C)CCn2c(cnc2CNc2cc(O)c(O)c(O)c2)C1 C1(C(=O)OC)CN(C(c2ccnc(OC(F)F)c2)=O)c2ccc(F)cc2O1 c1(CC)cnccc1CNC(=O)NOCCF CCCCCC(O)C(=O)N1CC2(C(N3CCC(C)CC3)=O)CCC1CC2 C#CC1CN(C(=O)C(CC=CC)NC(=O)CC=C)CCN1C C12(O)CCCN(C1)C(=O)CC1(CCC1)NC(=O)CC2.C(C)(C(=O)NC)=C(CC)C N1(C(CC2CC(=C)C2)=O)CCC2(CC1)CN(C(c1ncncc1Cl)=O)CC(C)O2 C1(C)(CNC(C(C)Cc2cnn(C)c2)=O)CCCN(C(=O)C2=CCSC2)C1 C1(NC(C(C)OCC)=O)CC(F)CN(C(c2cc(Cl)n(C)n2)=O)C1 C=C1CCN(C(=O)CC2CCOC2=O)C(C(N2CCN(C)CC2C)=O)C1 c1(C(=O)NC2(CO)CN(C(C3C(C(=O)OC)C3)=O)C2)cnc2ncnn2c1O c1(C(=O)NCCC2CN(C(C3CN(C)C3)=O)CC(C)O2)cccc2nccnc12 c1(C(N2C3CC(CC(NC(C(C)S(N)(=O)=O)=O)C3)C2)=O)cn2cc(F)ccc2n1 CCCC(C(=O)N1CCC(CNC(=O)CC2CCC3(CCC3)O2)CC1)S(N)(=O)=O N1(C(Cc2nc(C(C)C)sc2)=O)CC(NC(=O)C(F)(F)c2ccnn2C)CC1C Cc1[nH]c2ncccc2c1C(=O)N(CCNC(=O)Cc1cc(C2CC2)on1)C1CC1 C1(C(=O)NCc2ccc(OC)nc2)CC12CCN(C(=O)CCN=[N+]=[N-])C2 c1(C(=O)Nc2c(C(=O)OCC)cc(F)c(Br)c2)cc2c(=O)[nH]ccn2c1 Cc1nc(C(=O)NCC2(O)CN(C(C3CC4OC3C3CC43)=O)C2)c2ccnc-2[nH]1 C1(N(C(c2nc(CCC)oc2)=O)C)CC2CCC(C1)N2C(c1cc(CO)[nH]n1)=O N(C(=NCCC1CCOC1)NCCc1cccc(C)c1)C(COC)C CC1C(C(=O)N(CC2=CCSC2)C)CCN1C(C1CCC(C)(C)C1)=O C(=O)(CC(C)(C)CNC(c1ccn(C)n1)=O)NC(COC)CCO CC(C)(C#N)C(=O)NCCC(O)CNC(=O)C1=C(Cl)CC1 Cc1cc(NC(=O)CC2COCCN2C(=O)C(O)C(C)C)cnc1Cl C=CC(C)(CCOC)C(=O)NCC1(C)CC(NC(c2csnc2OC)=O)C1 N1(c2cc(CC)ncn2)CCOCC(NC(c2c(C(F)(F)F)coc2C)=O)C1 c1(C(=O)NC2CC3CN(C(CC4CC(=C)C4)=O)CC3C2)cnc2snc(C)c2c1 c1(C(=O)NCC2=CCN(C(C3OCC(C)(C)C3)=O)CC2)ccc2c(c1)C(=O)NC2 C1(O)(C(CNC(C2(CC(=O)OC)CC2)=O)C)CCN(C(=O)C=NOC)C1 c1(CC)nncn1NC(=O)C1CC(NC(c2cc3ccccn3n2)=O)C1(C)C C1(NC(C(C(=C)Cl)(C)C)=O)CC1C1CCN(C(C2CC3C=CC2C3)=O)CC1 c1(C(N2CC(NC(c3n(CC)ncn3)=O)C(O)C2)=O)c(O)cccc1Cl C=C(C)CC(C(=O)NC1CCC2(C(C)C)CC12)NC(=O)C(C(C)C)SC N1(C(c2scc(C)c2)=O)CC(F)CC1CN(C(=O)C(N1CCOCC1)C)C c1(CC)oc(C)cc1C(=O)N(CCCCCCNC(C1(C(=O)N(C)C)CC1)=O)C C(C(CC(=O)N1CCC(Cc2ccn(C)n2)C1)C1CCCCC1)OC N1(C(C2C(CC)C2)=O)CCC2(C(=O)NC3CC3C(C)C)CCCC12 C1(CC(=O)N(CCCO)CC#C)CCCN(C(c2nnc(S)n2C)=O)C1 C1(N(C(c2[nH]cc(C)c2)=O)C)CN(C(=O)COC2CC2)CCC1C Cc1noc(C)c1CCC(=O)NC(C1CCCCN1C(=O)Cc1ccnn1C)C N1(C(C(C)(C)C2CCOC2)=O)CC2(C1)SCCC2NC(=O)COCc1nc[nH]n1 CCC(CCOC)C(=O)NCC1CN(C(c2ccnn2COC)=O)CCN1C N1(C(CSS(C)(=O)=O)=O)CC(CNC(c2cnc(C3CC3)s2)=O)C2CC12 c1(C(=O)NCCOCCn2cc(-c3c(C)ncs3)nn2)c(C)nn(C)c1N C(=O)(C(O)(C(F)(F)F)C1CC1)NCCOCCCNC(c1c(C)ccnn1)=O N1(C(C(C(C(C)C)O)C)=O)CCN(C(c2cc[nH]c2)=O)C2CCCC2(C)C1 C1(=CC(=O)NCCN(C(=O)COC2(C)CCCC2)CCC)CN2CCC1CC2 N1(C(c2c(SC)csc2)=O)CC2CCCC2(CNC(c2cccc(O)n2)=O)C1 Cc1cc(C(=O)NCCC2CCN(c3ncccc3C#N)CC2)n2ncnc2n1 CCCC(C#N)C(=O)N1CCN(C(=O)CN(CC)CC)CC1C c1(C(N2C(CC)CN(C(=O)CC3CC(F)C3)CC2)=O)cc2c(s1)CCCNC2=O N1(C(Cn2c(C)ccn2)=O)CCN(C(=O)C(C(C)C)NS(C)(=O)=O)CC1CCO Fc1cccc2c1OCC2N=c1nc2scnc2c(NCCC(F)(F)F)[nH]1 C(=O)(C(C)(CO)CO)Nc1c(C(=O)Nc2ncn(C)c2)scc1 C1(NC(C2(OCC)CC2C)=O)C2CC3C1C3C2C(=O)NCCC1(CO)CC1 c1(C(N2CC3(CCN3C(c3ccsn3)=O)C2)=O)n[nH]c2c1CCCC2 C(Cc1ccccc1)(CC(=O)O)NC(c1n(C)cnc1)c1nnnn1C C1(C(=O)NC2(CC(=O)NCC(C)(C)F)CCC2)CC(=O)CC(=O)C1 c1(N2CCC(N(C(c3cc(C)[nH]n3)=O)C)C2)cc(CC(C)C)ncn1 C1(C(=O)NCC(C(C)C)NC(c2csc(-c3ccsc3)n2)=O)CC(C)(C)CN1C C(=O)(CC(CC)CC)NCC1(CNC(c2ncc(OCC)nc2)=O)CC(F)(F)C1 Cc1cccc(C(N2CC(N(C)C)C(CNC(C3(O)CC3)=O)C2)=O)c1Cl c1(C(=O)NCC2CN(C(COCC)=O)CC2C)ccc(C#N)cc1 c1(C(=O)NCCCC(C)NC(C(CC(=O)OC)(C)C)=O)ccc2c(c1)SCCN2 c1(C(=O)NCC(C)(CO)NC(C(C)OCCOC)=O)ccc(-c2cn[nH]c2)cn1 N1(C(CCn2ccc(C)n2)=O)C2CCCC1CN(C(C1CCCNS1(=O)=O)=O)C2 c1(OC)cn(CC(=O)NC2CCCCN(C(=O)C(O)C3CC3)C2)c(C)cc1=O C1(COC)CN(C(=O)Cc2ccc(C)o2)CCN1C(c1occc1F)=O C1(CSC)CCN(C(C2C=CCN2C(=O)CC2C=CCCC2)=O)C1 c1(NC2C3CN(C(CCSC)=O)CC2CC3)nc2ccc(C(F)(F)F)cn2n1 C1(C=C)(C(=O)NC(CC#C)C(=O)OCC)CCN(C(=O)CN2CCOCC2=O)C1 N1(C(C(CC)C)=O)CC2CCCN(C(=O)CCc3ccsc3Cl)C2C1 C(C)(CCCCNC(C1(CN(C)C)CC1)=O)NC(COCC(C)C)=O c1(C(=O)NC(C(=O)NC(CCCCC)C)C(C)(C)C)c[nH]c2ccccc12 N1(CCC(=O)N(CC(C)NC(=O)CN(C2(CC(C)(C)C)CC2)C)C)CCCCC1 N1(C(Cc2nc(CC)sc2)=O)CC(NC(c2ccc(Cl)cn2)=O)C(C)(C)C1 c1(C(N2CCC(COC)(NC(=O)COC3CC3)C2)=O)c2c(nn1C)CCCC2 N1(C(CCc2c(C)nccc2)=O)CCN(C(=O)C(C2CCOCC2)C)CC1CO c1(C(N2CCCN(C(CC(CC(C)C)C)=O)C(C)C2)=O)cccc2oc(O)nc12 C1(C(N(CCC(=O)NC(CC(=O)OCC)C)CC)=O)C2CC3C(C2)C13 CCC(O)CC(=O)N1CCC(O)(C(C)NC(C2CC2F)=O)C1 CC(C)(CCCNC(=O)CC1(n2cccn2)CC1)C(=O)NCC1CNC(=O)CO1 N1(C(C(OC)OC)=O)CCC(C2CC2)C1CNC(C1CC(N=[N+]=[N-])C1)=O N1(C(c2nc(C)oc2)=O)CCC(NC(=O)CC2CCC2)C(C)C1 c1(COC(NOCCCOCC)=O)cc2sc([N+](=O)[O-])cc2s1 c1(C(=O)NC2CCN(C(C(C(CC)O)C)=O)C2C)ccc2nc(C)nc(O)c2c1 c1(C(=O)NC2(C)CN(C(CN(CCCCCC)C)=O)C2)cnc(C(C)C)n1C C(=O)(C1=NOC2(CCC2)C1)N1CCCN(C(CC(CCSC)O)=O)CC1 C(=O)(C(C(C)C)c1cccnc1)NCC(C1CC1)NC(c1n(CC)ccc1)=O c1(C(N2CCN(C(c3c(C)cns3)=O)CC2CO)=O)cnc2[nH]nc(O)c2c1 c1(C(=O)OC)cc(OC)c(S(=O)(=O)NC(c2ccccc2)C2CCOC2)s1 c1(C(N(C(=O)NCCCC(O)OCC)C)C)ccccc1-c1cccnc1.CC C1(C)(C(=O)NC23CCC(CN(C(CCC#C)=O)C2)C3)C2CC3CC(C2)CC1C3 c1(C(N2C(C(N(CCOCC=C)C)=O)CCC2C(C)C)=O)ccc(O)c(C)c1 N1(C(C2CN(C)C2)=O)CC2(CC(C(=O)NCC(O)C(F)F)CO2)C1 c1(OC)ccc(C(N2CC3CC(C2)N3C(=O)CC2CCN(C)CC2)=O)c(Br)c1 C(C(C)(C)CC(=O)N(C)C(c1ccc(C(F)(F)F)cc1)C)OC N1(C(C2N(CCC)CCCC2)=O)CCC(F)(C(=O)OC)CC1 C1(O)(CNC(c2[nH]cc(C)c2C)=O)CCCN(C(c2cc(Cl)cnc2O)=O)C1 N1(C(c2cccc(C#C)c2)=O)CCC2CN(C(=O)C=Cc3cn(C)cn3)CC2C1 N1(C(C=CC)=O)CCC2(COC(CNC(c3cccn3C)=O)C2)C1 N1(C(C2CCC(C)(C)O2)=O)CC2(C1)CN(C(=O)CC1=CCCC1)CC2CO c1(C(N(CC(C)CNC(=O)CC=CC(C)(C)C)C)=O)cnc2c(c1)OCCN2 N1(C(C2CC(=C)C2)=O)CCC(NC(=O)C(F)Cc2ccccc2)C1(C)C c1(-c2cc(NC(c3c(O)cccc3F)=O)sc2)ccc(B(O)O)cc1 N1(C(c2cc(CC)no2)C(=O)NC(C)C)CCCC(c2nncn2C2CC2)C1 C1(CC(=O)NC2(CNC(c3scc(COC)c3)=O)CC2)CCc2sccc2C1=O C1(C(=O)NC2(C(N3CC(F)(COC)C3)=O)CCSC2)(N(C)C)CCCSC1 C1(c2nnnn2C2CCOCC2)(OCCNc2ccccc2)COC2(COC2)C1 Cc1n[nH]c(C)c1CC(=O)NCC1C=CCN1C(c1cc(C2CCC2)[nH]n1)=O CCCC(CC(=O)N1CCCC(C2OCCO2)CC1)c1ccccc1.C1C(=O)N1 c1(COCCN(S(Cc2c(C)ocn2)(=O)=O)C)ccccc1Br c1(CC)cc(C(=O)NCC#CCNC(=O)Cc2csc(Br)c2)ccc1F C1(C(N(C)CC2CCC(=O)N2)=O)CCC2(CC2)N1C(C1CC2CCC1CC2)=O C1(F)(CNC(C=CC(=O)N(C)C)=O)COCCN(C(C2C3(CC3)C23CC3)=O)C1 N(S(=O)(=O)N(C)CCc1csc(C(F)F)n1)CCNC(=O)OC(C)(C)C c1(CC(N2CC(NC(C(c3ccccn3)C)=O)C2)=O)ccc(Cl)nc1 c1(OC)cc(C(N2CC(NC(=O)C(C)(F)F)CC2C)=O)c(N)cc1F CC1COCC(C(N2CCOCC2CC(=O)NC(c2ccccc2F)C)=O)O1 c1(SCCC(=O)NCC2(COC)CN(C(=O)CSC)C2)ccccc1Cl Cc1cc(Cl)ccc1NC(C1CCCCC1NC(=O)CCC1CCC(=O)C1)=O c1(C(N(C2C3CN(C(C(CSC)(C)C)=O)CC32)C)=O)coc(=O)c2ccccc12 c1(C(N2CC(CNC(CCNC(=O)NC)=O)C2)=O)cnc(O)n1CC N1(CC(COC)(C)O)CC(C(=O)OC)CC(CNC(=O)OC(C)(C)C)C1 c1(C(N2CC=C(CNC(C3CCC4(CC4)C3)=O)CC2)=O)cnn2c1CCCC2 N1(C(CNC(=O)NC)=O)CC(C(=O)NC(C)Cc2nncn2C)CC(C)C1 C1(CCC=C)(C(=O)NC(CC(=O)OC)C2CC2)CN(C(c2ncsc2NC)=O)C1 C=CCC(C)(C)CC(=O)NC1CC2CC(C1)N(C(c1cn3ncccc3n1)=O)C2 N1(C(CC)=O)CCC(C2CCN(C(c3cnn(CC(F)(F)F)c3)=O)C2)C1 C1(NC(CSC)=O)COC2(CCN(Cc3scnc3C)CC2)C1 CCC(CC(=O)N1CCCCC1C1(NC(c2oc(C)nc2C)=O)CC1)C1CCC1 C1(NC(COCCNC(C(COC)(C)O)=O)=O)CCCCNC1=O N1(C(C2C(OC)(OC)CC2)=O)CCC(C)(CCNC(C2CCCS2(=O)=O)=O)CC1 C(CC(CC)(CC)NC(=O)COc1cnn(C)c1)NC(COCCCC)=O C1(CC(=O)NC(C(C)NC(CCCOC(C)C)=O)CO)C=NN(C)C1=O CN1CCC(C)(C(N2CC3CC(NC(C4CC(=O)NC(=O)N4)=O)C3C2)=O)C1=O C1(NC(=O)CCc2ccoc2)CCC12CCN(C(=O)CC(F)(F)C(F)(F)F)CC2 Cc1conc1C(=O)NC(C(=O)NC1(C(C)C)CC1)C1CCCO1 N1(C(C(CC)(F)F)=O)CC(C2CCN(C(C3(CO)CCCCO3)=O)CC2)C1 c1(C(N(C2CC(NC(c3ccc(F)o3)=O)C2)C)=O)ccn(CC(F)F)c(=O)c1 c1(CC(=O)NCC(C)N(C(=O)CN(C)C)C)csc(-c2ccccc2)n1 C(=O)(CCCCN1CCCCC1)NCC1(O)CC(CNC(c2n(C)ccn2)=O)C1 N(C(=NCCSC)NCc1c(F)cccc1Cl)C1CC(OCC)C1(C)C CC1CCCCC1OCC(=O)NC(C)(C)CCCNC(=O)CC1(C)CC(F)(F)C1 CC1CN(C(c2nncs2)=O)CC(C)CN1C(c1cc2ncccc2[nH]1)=O N1(C(c2cc(-c3ccc(C)s3)on2)=O)CCc2nc(=N)[nH]cc2C1 C1(OC)CC(C(=O)NCCC2CCCN2C(c2ncsc2C2CC2)=O)CC1OC C1(C(F)(F)F)(C(N2CC(CCCCNC(COCC#C)=O)C2)=O)CCCCC1 CC1(C)CC(C(=O)NCC2(C)CCCN(C(=O)Cn3ncnn3)C2)CC1(C)C c1(C2N(C(c3scnc3Cl)C(=O)NCCCCCC)CCC2)cc(F)ccc1F c1(C(=O)NC2(CNC(C(CC)C#N)=O)CCCC2)cccc2c1CCCC2 c1(OCCCNC(C2(N(C)C)CCOC2)=O)cccc(CC#N)c1 N1(C(C2C(OC)CCC2)=O)CCN(C(=O)C=Cc2ccccc2C#N)CC(O)C1 C(=O)(CS(=O)(=O)CC(=O)OC)N1C2CCC(NC(C(C=C=C)C)=O)(CC2)C1 O=C(C#CC1CCOC1)NC1CC2CC1N(C(=O)C1=CCCC1)C2 C1(F)(CNC(C(CC)CC)=O)CCN(C(=O)CC2CCC(F)(F)CO2)CC1 c1(-n2cc(-c3cccc(C)c3C#N)nn2)ccc(S(=O)(=O)CCN(C)C)cc1 C1(CNC(C2N(C(C)(C)C)CC2)=O)C=CCN1C(c1cc(C(N)=O)c[nH]1)=O Cc1ccc(S(=O)(=O)NCCC(=O)N(C)CCNC(=O)C(C)CN(C)C)cc1 Cc1ncc(C(N2CCCCC(CNC(C3CCCC3C3CC3)=O)C2)=O)c(=N)[nH]1 CCC(CO)NC(=O)N(C1CC(CO)C1)C1CC1 C1(CNC(c2cn(CC=C)nn2)=O)CCCN(C(c2cncc(F)c2)=O)C1 C1(C(=O)NC2(CCOCC)CCCC2)CN(C(=O)C=C(C)C(C)C)C2(CCC2)C1 N1(C(CNC(=O)OC)=O)CCCC(O)(CNC(C2(C(C)C)COC2)=O)C1 N1(C(C2CCC(C)O2)=O)CC2(NC(=O)CCC(C)(C)F)CCC1CC2 C1(NC(c2c(C(=O)OC)[nH]cc2)=O)CCCC(NC(C2CCCS2)=O)C1 c1(-c2cn(CC3N(C(C(n4c(C)ccn4)C)=O)CCC3)nn2)ccc(CO)cc1 C1(NC(C2C(CC)CCN2C(=O)CC2CC(C)(C)CO2)=O)CCCCN(C)C1=O Cc1csc2ncnc(N3CC4(CCN(C(=O)C(O)C(C)C)C4)C3)c12 CC1(C)CCCN(C(C2CN(C(c3cc(O)cc(F)c3)=O)CC(C)(C)C2)=O)CC1 CC(C)C(CC(=O)N(C1CCSC1)C)NC(c1cc(C#N)cn1C)=O C1(CC=C)(NC(=O)CCC#CC)CCN(C(=O)CSC2CCOC2=O)C1 C1(NC(=O)CC2CC3(CC3)C2)C2CCN(C(c3c[nH]nc3C3CCC3)=O)CC12 c1(C(N2C(C)CCC(NC(C3CC4(CSC4)C3)=O)C2)=O)cnc2cccnc2c1 C1(CN(C(=O)CCC(=O)NC2CCSC2)C)CCC(C(=O)Nc2nccs2)CC1 c1(C(=O)NC2C(CNC(CN(C(=O)OC)C)=O)CC2)cncc(C(C)(F)F)c1 C(c1ccccc1)=CC(=O)NC1CC(C(N2CCCC(C(F)F)C2)=O)C1 Cc1c(C(=O)NCC2CCCN(C(=O)COC(C)(C)C(F)(F)F)C2)cccc1N C1(C(=O)NCC(CCNC(C(CC(=C)C)OC)=O)OC)Cc2ccccc2S1 C1(C(=O)NCC(N(C)C(c2ncc(C(F)F)s2)=O)C2CC2)CC2CCCCN2C1 c1(OC)sccc1C(=O)NC(C)CN(C)C(c1cnc(Cl)[nH]1)=O N1(C(c2ccc(CNC(CC(COC)C)=O)cn2)=O)CCC(OC)C(C)(C)C1 c1(OC)ccc(SCCC(=O)NC2COCC2NC(C2CSC2)=O)cc1 c1(C(N2CCC(NC(c3cncc(CC)c3)=O)C2)=O)ccc(F)c(Br)c1 C(=O)(CCCC(=O)NCCCCCNC(=O)Cc1ncc(Cl)s1)OC(C)(C)C c1(CNC2C(C(=O)NC(CC)C)CCC2)cccc(-c2cccc(Cl)c2)c1 C#CCC(CC#C)C(=O)N1CCCC(CCNC(=O)CCOc2cccnc2)C1 C(=O)(C(CC1CCOC1)CNC(=O)O)NCC.C(C(=O)N(C(C)(C)C)C)N(C)C CS(=O)(=O)c1cc(C(N2CC3CC2(CNC(=O)COC2CCCOC2)C3)=O)co1 c1(OC)cncc(C(=O)NCCC2CCCN2C(=O)COCC2CCOC2)c1 c1(C(N2CCC(N(C)C(c3cnsn3)=O)C2)=O)cc(Br)cc(F)c1F c1(CC(=O)NC2CC2NC(C2C=CC=CC=C2)=O)cc2nc[nH]c2cc1Br C1(NC(CCc2cccc(C)c2)=O)CC2CN(C(C3(O)CCCC3)=O)CC2C1 C1(CNC(c2c(CC)cc[nH]2)=O)CN(C(c2nc(C)n(C)c2C)=O)C(C)(C)C1 CC1N(C(c2c(CNC(c3ccon3)=O)nnn2C)=O)CCC1(C)C C(=O)(C1CCCc2scnc21)NCCC(CNC(=O)CC1(O)CCC1)O c1(NC(C2(C(=O)OC)CCNC2)=O)ccc(CC2(O)CCNCC2)cc1 CC1(C)CCCOC1C(=O)NCC(c1ccccc1)NC(=O)C1=C(Cl)CCC1 C(=O)(C1c2c[nH]nc2CN1C(c1cccc(CO)c1)=O)NCC(CC(=O)OC)O c1(C(c2nnnn2Cc2ccccc2)NC(CSC)(C)C)nc(C(F)(F)F)cs1 C(C)(CNC(C1(O)CCC1)=O)(C(C)C)NC(c1cnc(C(C)OC)s1)=O C(=O)(C(CC(C)C)C(C)C)NCC(CNC(C(COC)OC)=O)(C)OC C1(N(CCCC)C(c2cc(OC)n[nH]2)=O)CCN(C(=O)C(C)NC(C)=O)CC1 C(=O)(C(O)Cc1cnc[nH]1)NC(CN(C(CCC)=O)C)CC N1(C(C2CCC3(CCC3)C2)=O)CC2CCN(C(=O)C(F)(F)CO)CC12 c12cccnc1C2.CC1CCC(C(=O)NCc2cn(Cc3cccs3)nn2)O1 CC1(C)CC(NC(=O)C(C)(F)C(C)(C)F)CN(C(c2ccccc2)=O)C1 c1(C(=O)NC2CN(C(C(C)C3CCCC3)=O)CC(F)C2)cnc2[nH]cnc2c1 N1(C(c2c(C)scc2)=O)CC(NC(C23CCC2CC3)=O)CC12CCC2 C1(C(=O)NC2CC(NC(C3C(C(=O)OC)CC3)=O)C2)CCCCC12CCC2 Cn1[nH]c(C2CC(CNC(=O)CNc3ccccc3C#N)C(O)C2)nc1=O C(C)(CCCN=c1[nH]c(=NC2CN(C)C3(CCC3)C2)[nH]c2cccnc12)OCC C1(C(=O)NCc2ncc(C)nc2)CN(Cc2ccc(O)cc2)CCC1O c1(OC)cccc(C(=O)NCc2ccc(N(C)C)c(F)c2)c1OOC(F)F C1(NC(C2N(CC)CCC2)=O)CN(C(=O)C(C)(C)n2ccc(C)n2)CC1F C1(CNC(C(CC=C)NC(C)=O)=O)CC2CCC1N(C(c1cc(Cl)no1)=O)C2 Cn1oc(C(N2CCC(c3cn(C(c4ccccn4)CCl)nn3)CC2)=O)cc1=O C(=O)(C1CCCc2ncccc21)N1C(CNC(C2(COC)CCCO2)=O)CC1 c1(C(=O)NC(CC)CNC(C2CC3CCCC(C2)C3)=O)ccc(F)cc1[N+](=O)[O-] N1(C(C2C(CCC)C2)=O)CC2CCC2(CNC(c2cnc(S)n2C2CC2)=O)C1 N12CC3CCC(C3C1)Nc1nccc(n1)CC2=O.C(C(=O)OC)=CCOC C(=O)(C1COc2ccc(Cl)cc21)N1CCC2(OCCN(C(C3CC3(F)F)=O)C2)C1 c1(C(N2CCC(NCc3ccc(C)c(F)c3)C2)=O)c[nH]c2cc(C#N)ccc12 CCCCC(C(=O)NC(C)CCCNC(c1ccnc(F)c1OC)=O)C(C)C C1(C#N)(C(N2CCC(NC(CC(CC)OC)=O)CC2)=O)CCC(=O)CC1 c1(-c2cn(C3CCN(C(=O)CCn4ccnn4)CC3)nn2)ccc(I)c(Cl)c1 N1(Cc2nnc(C)s2)CCC2(CC1)CN(C(c1ncn(C(C)C)n1)=O)CC(C)O2 C12(CCn3cc(CCCC)nn3)CCC(CC1)N(C(=O)C(CC(C)C)OC)C2 CCCCCC(F)C(=O)N(CC(O)CNC(c1ccc(CNS(C)(=O)=O)o1)=O)C C(C(C)(CNC(c1cncc(CNC(=O)CCCn2cccn2)c1)=O)CO)OC Cc1nc(=NCC2C(C)CCCN2C(=O)Cc2ccc(F)cc2F)c(C#N)c[nH]1 C12CN(CC1CC)C2=O.C(C(O)C(=O)NC)NC(C=CC=CC)=O N1(C(CCOCCN(C)C)=O)CC(CC(=O)NCc2n[nH]cc2CO)C2(CC2)C1 N1(C(c2ccc(C)cn2)=O)Cc2ccccc2C(NC(=O)CC2COC(=O)C2)C1 C1(NC(C2CC3C=CC2C32CC2)=O)CN(C(=O)CC2(O)CCC2)C2(CCOC2)C1 CC1=C(C(=O)NC2CC(C(N3CC(C(N)=O)C(C)C3)=O)C2)CCC1 O=C1CCN(CCC23CCC(CC2)CC3)C(=O)N1Cc1ccccc1C(F)(F)F C1(CNC(=O)Cc2ccccc2F)CCC2(CCC2)C1NC(=O)C1CC1 Cc1ccc(NC(C2(CNC(C3CC(=O)C3)=O)CC23CCC3)=O)cc1O c1(C(=O)NCC2OCCC(NC(C3N(N=O)CCC3)=O)C2)cc2n(n1)CCCN2 C(=O)(CCCCCC#N)N1CCCC(C)(CNC(c2nc(C(C)C)oc2)=O)C1 c1(CNC(C(C)SC)=O)cc(O)nc(CNC(c2cccn2CC2CC2)=O)n1 C(CCC(C)(F)F)CCN1CCC(C2N(C(c3ccccc3)C(C)C)CCC2)C1 CC1(C)CN(CCC2=CCCCC2)CCC1NC(=O)Cc1ccc(Cl)s1 n1(CC)ncc(C(=O)NC(C)CNC(=O)CCC2CC(C)(C)CO2)c1C1CC1 N1(C(C(C(C)C)O)=O)CCCC2(C1)CN(Cc1ccnn1-c1ccccc1)C2 C(=O)(C1CCCc2nn[nH]c21)N1CC(NC(C(C)=C2CCCC2)=O)CC12CCC2 Oc1ccc2c(c1)C(Nc1ncc(C3CC3)cc1Br)CCC2 c1(CC(=O)NCCCC(CCC)NC(C(CC=C)C)=O)noc2ccccc12 c1(C(=O)NC2CN(C(c3c(SC)cccc3)=O)C(C)C2)cc(F)c(F)c(F)c1F N1(C(C=CCOC)=O)CC2CCN(C(c3cnc(C(C)C)nc3C)=O)CC(C2)C1 C1(NC(C2N(CC#C)CCC2)=O)CN(C(=O)C(C)OCC2CC2)CC1C N1(C(C(C)CN)=O)CCn2c(nc(C(N3CC(O)CC(F)C3)=O)c2Cl)C1 C(=O)(CC(C)(C)C(C)=O)NC(CCC)C(N1CCCCC(N2CCC2)C1)=O C12(N)CC3CC1C2C3.C1(CC=O)CCC1NC(=O)C(=O)NCC1CC1 C1(NC(C(c2n(C)ccc2)=O)=O)CC2CC(NC(C3CCC(=O)N3)=O)CC2C1 CCC(C)(C)C(O)C(=O)NC1CCN(C(=O)Cc2ccc(S(=O)(=O)NC)s2)C1C N1(C(c2c(C)onc2)=O)C2CCC1C(F)C(NC(=O)CCn1ncn(C)c1=O)C2 O=C(CCC1CCC1)N=c1ccn(CC(=O)NCC2CC3C=CC2C3)c(O)n1 C1(CNC(C=C=C(C)C)=O)CCN(C(=O)CCCC2CCC2)CC1(F)F C1(C(=O)NCC(CN(C(CSc2ccc(C)cc2)=O)C)O)OCCOC12CCC2 CC1(C)CN(C(=O)COCC(F)(F)F)CC(CNC(C2(CO)CCCO2)=O)O1 C1(C(N2CCCCC(NC(C3CCC(=O)C3)=O)C2)=O)CC2CCCC(C1)C2 CC1CC(NC(c2cc(-c3ccncc3)on2)=O)CN1C(C1CCCCO1)=O C(N=c1[nH]c(Cl)ncc1Br)C1C(C(F)(F)F)CCN(C(CC2CCC(=O)NC2)=O)C1 C12(C(=O)NCC3(OC)CN(C(COc4cn(C)nc4)=O)C3)CCCCC1C2(F)F C1(NC(C2(C)CCCCC2)=O)Cc2ccccc2C1NC(=O)CC1(C)CC1F N1(C(c2nc(CCCCC)sc2)=O)CC=CC(NC(=O)C(C2CCC2)OC)C1 C(C(CC1CC1)C(=O)NCC(=O)NC(C)(C)C)NC(c1ccc(C)o1)=O c1(NC(c2n(C(CC)C)nnn2)c2ccn(C)n2)cccc(NC(=O)C(C)C)c1 N1(C(Cc2cc(C)sc2)=O)CCC(CF)(NC(=O)C(CCO)N(C)C)C1 Cc1cc(C)n(CCCNC(=O)CC2CCN2C(C2CSC2)=O)n1 c1(C(=O)Nc2cccc(NC(COCCOC)=O)c2)nncc2c1CCCC2 c1(CN2C3C(C(N4CCC(N5CCCC5)CC4)=O)C(C3)C2)cc(F)c(Cl)cc1F c1(C(=O)NC2CC(CNC(C3(c4nccs4)CC3)=O)C2)cc(Cl)c[nH]1 c1(C(=O)NCc2c(CCNC(CC(COC)C)=O)ocn2)cc(C)c(Cl)cc1F c1(C(=O)NC2C(CNC(C(CCOC)C)=O)CC2)ccc2c(c1)C(=O)NC2 C1(C(=O)NCc2cc(OC)no2)CCC2CCC1N2C(=O)C1=CCCC1 NS(=O)(=O)CCCC(=O)NCC(F)CNC(=O)CSCc1ccncc1 CCC(C)C(C(=O)N1CC(OC)C(c2cn(-c3ncc(C)s3)nn2)C1)OC C1(CNC(C(C)(C)C2CCCC2)=O)CCC2(CN(C(C3CC(F)C3)=O)C2)O1 Cc1scc(C(=O)NCC(C(=O)NCCc2ncon2)N(C)C)c1C c1(NC(C2C3(CN(C(C(C)(C)C)=O)C3)C2)=O)cnc(Cl)cc1Br N1(C(c2cnc(CC)o2)=O)CCCC2C(NC(=O)Cc3cncn3C)C(C)(C)C12 N1(C(C2CCC(NC(c3c(C)cns3)=O)CC2)=O)CC2OCCN(C)C2C1 CCC(C)(CO)C(=O)NCC1(CNC(c2ccc[n+]([O-])c2)=O)CCCCC1 C1(N(C(c2c(CC)csc2)=O)C)CCN(C(=O)CCN(S(C)(=O)=O)C)CC12CC2 C#CC1(NC(=O)NCC(c2nc(C(C)C)cs2)OC)CCCC(C)(C)C1 CC(C(=O)C(=O)COCC(F)F)=CCNCC=CCN N1(C(CC(C)(C)SC)=O)CC2(CNC(c3cnc(C)nc3)=O)CC1CCO2 CCCC(CNC(=O)CCC=Cc1cccnc1)C(=O)NOCCOCC C12(C(=O)NCC(c3cccc(Br)c3)(C)C)CC1CN(C(c1nc(Br)cs1)=O)C2 N1(C(=O)NC(c2cc(Cl)cnc2F)CC)CCSC2COCCC12 C(=O)(C#CC1CCOC1)NC1(CN(C)C(C2(c3ncccc3F)CC2)=O)CC1 c1(CNC(c2c(OC)cc(Br)cc2)C)cc2c(nc1O)CCN(C)C2 c1(C(N2CC(CCNC(C(CC)C(=O)OC)=O)C2)=O)ccc(Cl)c2ncccc12 c1(C(N2CCC(CCNC(Cc3ccn(CC)n3)=O)C2)=O)cnncc1NC c1(NC(C2(NC(C(F)=CCC)=O)CC2(C)C)=O)ccc[n+]([O-])c1 c1(C(=O)Nc2c(C(=O)NC(c3ccccc3F)C)n[nH]c2)cc(Cl)nc(Cl)c1Cl C#CCC(C)(CC)C(=O)NCCSCC(N1CCCC(OCCC)C1)=O C1(CC(=O)N(C2CN(C(C3CCOCC3)=O)CC2O)C)CCC(C)(O)CC1 c1(OC)cccc2c1OCC(C(=O)NCCCc1cn(C3CCOC3)nn1)C2 C1(C(=O)NCC(CNC(C2C(CCC)CCC2)=O)(C)C)(COC)CC2(CCC2)C1 N1(C(CCc2nc(C)sc2)=O)CCC(CNC(c2cnn(CCO)c2)=O)C(C)C1 N1(C(C2CC=CC(NC(c3n[nH]c(C)c3C)=O)C2)=O)CCC2(CNC(=O)C2)C1 N1(C(C(C)C2CC2)=O)CC2CCC1C(CNC(c1coc(S(C)(=O)=O)c1)=O)C2 CC1(C)CC(C(N2CCC3C(NC(=O)CSC(F)(F)F)C23)=O)CCO1 N1(C(=O)CCc2cnc(O)[nH]2)CC2CCCC(C1)N2C(=O)C(CO)C(F)(F)F N1(C(C2CC(Cl)(Cl)C2)=O)CCC2CCN(C(c3ccsc3)=O)C2C1 C(CCCC(CO)NC(C1CC2CC2C1)=O)NC(CCc1c(C)nn(C)c1)=O c1(CC)c(C(=O)NC(C)C(CO)NC(c2ccsn2)=O)cnn1CC(C)C c1(C(=O)NC(C)CCCNC(=O)Cc2cncs2)ccc2nc(CO)[nH]c2c1 N1(C(c2c(SC)nccn2)=O)CCCC2(CCN(c3ccnc(C#N)n3)C2)C1 c1(C(N2CC(C(C)NC(c3nnc(S)n3C)=O)C2)=O)c(F)ccc2[nH]ccc12 N1(C(C(F)OC)=O)CC(NC(C2(C)CNC(=O)C2)=O)CC2(CC2)C1 C12(NC(CCCOC(C)(C)C)=O)CCC1CN(C(=O)CC1(O)CCOCC1)C2 C(=O)(C1CCc2ccccc21)NC1C(C)CN(C(=O)CC(O)CN(C)C)C1 c1(C(N2CCN(C)CC2C)C(=O)Nc2c(CC)cccc2)cc(S(N)(=O)=O)cs1 C1(OCC)(CNC(=O)CC2CCCC2)CN(C(C2CC2Cl)=O)C1 c1(NC(C(CNC(c2[nH]cc(C(C)=O)c2)=O)O)=O)cc(CO)cc(C)c1 N1(C(CCOCC#C)=O)CC(C)(C)CC1CC(N1CCN(C)CC1CO)=O C1(CC(=O)NC2CCN(C(C=CC=CCC)=O)C2C(C)(C)C)CC2(CCC2)CO1 Cc1ccc(F)c(CN2CC=CC2C(=O)Nc2ccc(Cl)c(O)c2)c1 CCCCCCC(CC)C(=O)NCCCN(C(=O)C(F)C(=O)OCC)C CC1(CC(=O)NCC2CCOC2C(N2CCC(C(F)F)C2)=O)CCOC1 N1(C(C2CC3(CC3)C2)=O)CC(C2CC2)(C(N2CC3CC3C3CC23)=O)C1 n1(SCC(=O)NC(CC)CN(C(=O)C(C)Sc2ccncc2)C)ccccc1=O C(C(C)(O)CNC(=O)CC1(C2CC2)CC1)NC(CN(C1CC1)CC)=O CC1CC(n2nc(-c3ccccn3)nc2C(C)CCc2cccc(Cl)c2)CCO1 C12(C(N(C)Cc3c(CNC(C(C)OCC)=O)cccc3)=O)CCCN1CCC2 c1(C(N(C2CN(C(Cc3ccc(SC)cc3)=O)C2)C)=O)cn2c(n1)CCCC2 C1(CNC(C23CC(CCC)(C2)C3)=O)CN(C(=O)CSC(C)C)CCC1(C)C c1(CC(=O)Nc2cc(CO)ccn2)cccc2ncccc12 CC1(C)CCC(c2nnnn2C2CC2)(NCc2cn(-c3ccccc3Cl)nn2)C1 c1(NC(C2CC(C)(N=c3[nH]ncs3)C2)=O)ccc2c(c1)NC(=O)C1CCCN21 c1(C(N2CCC(CC(=O)N(C)Cc3nc[nH]n3)C2)=O)cnn(C(C)(C)C)c1N Nc1c(C(N2CCN(C(=O)CO)CC2)=O)cccc1I C1(NC(C(CC=C)(C)NC(C)=O)=O)CCN(C(=O)C=CCF)CCC1CO c1(C(=O)NC(C2CCN(C(=O)C(C)(C)CN(C)C)CC2)C)ncc2[nH]ncc2n1 C1(C(=O)NCC(C)NC(CCCC(C)C)=O)CCCC2(CCC(F)(F)CC2)O1 Cc1scc(C(=O)N(C)CCNC(=O)CCC2CCC(=O)N2)c1Br S(=O)(=O)(c1ccc(N2CCC(CN(C)C)C2)c(F)c1)NCCN(CCC)CCC Cc1ccc(CC(=O)NC(C)(CNC(C2CCC2(C)C)=O)CO)s1 C1(C(N2C(C=CC(=O)NCCC3OCCO3)CCC2)=O)CC2(CCCO2)C1 C1(NC(c2c(C)ccs2)=O)CCN(C(c2cc(-c3cnn(C)c3)no2)=O)CC1O C(C(C)(C)CNC(C1(CNC(=O)CC(C)O)CCC1)=O)OC C1(NC(c2nnn(CC)c2C)=O)CCN(c2nc(Cl)ncc2C)CCC1CO c1(C(=O)NC2CCN(C(=O)CCc3cccnc3)CC2F)cnn2ccccc12 c1(OC)ccccc1C(N)CC(=O)NCC1CC1c1ccc(O)cc1 C1(NC(=O)C2=CCC2)CC2CCC(C1)N2C(c1c[nH]nc1C1CCCCC1)=O C1(CCNC(c2c(OC)nccc2C)=O)CN(C(=O)C(O)C2CC2)CCS1(=O)=O Cc1c(NCC(C)CC(C)C)nc[nH]c1=NCC1CC2(C1)C(F)(F)C21CC1 C1(C(N(C2(C(=O)NCC3CCCCC3)CC2)C)=O)CCCN1C=O C1(C(N2CCC(C(=O)OC)C2C)=O)CN(C(=O)Cc2cc(C)cs2)CC12CCC2 C1(C(N(C)C)=O)CC(F)(F)CN1C(c1cccc(N(C)C)c1)=O c1(C(N2CCC(CNC(CC(C(=C)C)O)=O)CC2)=O)cc(F)c(Cl)c(N)c1Cl C(=O)(C1=C(Cl)CCCC1)NCC1(F)CCC(CNC(C(=O)N(C)C)=O)CC1 C1(C)(C(N2CCCC(CCC(=O)NC(CC)C(=O)NC)C2)=O)CCC2CC2C1 N1(C(C(CCC)C)=O)CCC(C(C)C)CC1CNC(c1ncoc1C(C)(C)C)=O C12(CNC(CCCC#C)=O)CC(CO1)N(C(C1(C)CC=CC1)=O)C2 C(N=c1cc(C#N)nc(C2CC2)[nH]1)C1(NC(C2CCCC(C)C2)=O)COC1 Cc1c(CNC(c2n[nH]cc2NC(C2CC3CCC2C3)=O)=O)cnn1C Cc1ccc(-c2nc(NC(=O)C(=O)NCC3CC(=C4CCC4)C3)sc2C)c(C)c1 N1(C(C)=O)CC(C)CN(Cc2cccc(C(F)F)c2C)CC1C C1(NC(=O)C(O)c2ccco2)C2COCC1CN(C(=O)C(N1CCOCC1)O)C2 N1(C(C=CCOC)=O)CCN(C)C(CNC(c2ccc(C)c(F)n2)=O)C1 C(=O)(C(O)P(C)(C)=O)NC1(COC)CCN(C(c2csc(-c3nc[nH]n3)n2)=O)C1 Cc1cncc(C(=O)NC(C(=O)N(C)Cc2occc2C)C(C)C)c1 CC(C)C(CC(=O)N1CC(C)=C(C)C1)NC(c1nc[nH]n1)=O CC(C)(C#N)C(=O)NC1CCN(C(c2cnc(-c3cnccn3)s2)=O)C1 CC(N=c1nnn(C)[nH]1)C1CCCCN1C(=O)Cc1cccc(Cl)c1F Cc1c(C(=O)NCC2CCN2C(=O)CCCCC(F)(F)F)oc2c1C(=O)CCC2 C#Cc1ccc(Cl)c(C(=O)NCC2(F)CCN(C(C3CCCOC3)=O)C2)c1 CC1N(C(C2CC(O)CN2C(C2CC(F)CN2C)=O)=O)CC(C)OC1(C)C N1(C(c2c(C)onc2)=O)CCC(CNC(=O)Cc2ccc(Cl)c(Cl)c2)C(C)C1 C(=O)(CCC=CC(C)C)NC1C(NC(C2(C(=O)NC)CC2)=O)C1 C1(S(C)(=O)=O)(C(N(C2CN(C(=O)C3=NOC(C)(C)C3)CC2O)C)=O)CCCCC1 c1(C(=O)NC2CCN(C(c3c(C)n(C)nc3)=O)CC2C)c(F)ccc(F)c1F N1(C(Cc2cc(C)on2)=O)CC2CC(C(=O)NCc3ccc(O)cc3C)C(C2)C1 C#Cc1ccc(C(=O)N(C2CC(NC(=O)CC3(C)CC3)C2)C)c(OC)c1 C1(C(=O)NC2(CCC(=O)NC(C)CC3(O)CCC3)CCCC2)CC2(C1)CC21CC1 C1(COC)CN(C(=O)CCc2cccc(OC)n2)CCN1C(=O)C(C)C1CCC1 C1(NC(N2C(C)CCC(C(=O)OC)C2)=O)CCc2cnn(C)c2C1 c1(C(N2CC(CCCNC(C(C)N(C)C)=O)OCC2)=O)c(O)cccc1F S1(=O)(=O)c2cccc(c2)C(=O)N1C.C(CCCC(=O)NC(C)(C)C)NC(CC)C C#CCCCCC(=O)NCC1CCN1C(C1CCN(C)CC1)=O N1(C(CN2CCN(CC)C(=O)C2=O)=O)CC2CC1CN(C(C1(N(C)C)CC1)=O)C2 C1(c2n(C(C)(C)C)nnn2)(NCCCn2cncn2)CCC2C3CCC(C3)C12 N1(C(C(C(C)C)F)=O)CC(NC(=O)CSCc2ccc(F)cc2)CC12CCCC2 C(=O)(C(C)(O)C(C)C)NCCNC(c1c(CC(=O)OC)cccc1)=O CC1(C)C(CNC(c2cc(Cl)sc2Cl)=O)CCN1C(=O)C=Cc1nccs1 CON(CCC(=O)N(C(C)C(C)C)C)C(=O)c1cccc(C)c1F N1(C(COCC)=O)CC(c2ccc(Cl)cc2)N=C1N1CCN(C(C)=O)CC1C c1(C(N2CCN(C(CS(CC)=O)=O)C(CF)C2)=O)ccc(C(C)C)cc1[N+](=O)[O-] C(=O)(C(C)C1=CCCC1)NC(CC=C)CNC(c1ccn(C)c1C)=O C(=O)(C1=C(F)CN(C(C2CC2(C)C(C)C)=O)CC1)NCCCC(=C)C Cc1ccc2ncc(C(=O)NCC(C)CNC(=O)CC3CC3C3CC3)n2c1 C(=O)(C(CC(F)F)N(C(=O)C=CC1CCCN1C)C)NC(C)CC(C)(C)C N1(C(C(C2CC2)SC)=O)CC(C(=O)N(C2CSC2)C)CCC1(C)C c1(NC(C2CCC(C(N3CC(O)C(F)C3)=O)C2)=O)c(Br)ccnc1Cl N1(C(C2C(C)(C)C2)=O)CCCC2(CC(NC(c3c[nH]ccc3=O)=O)C2)C1 C1(NC(C(COC)C)=O)CCCCC12CCN(C(C1CSCCS1)=O)CC2 C1(NC(CCC2(NC(c3cnn(C(C)C)n3)=O)CCC2)=O)CN2CCC1(F)CC2 N1(CC)CC2(CCN(C(c3cc(C(F)(F)F)ccc3O)=O)CC2)CNC1=O C1(O)(C(=O)NCCN(C(=O)NC2CCCCC2)CC)CCSC1 C(S(=O)(=O)c1ccc(Cl)c(Cl)c1)c1ccc(CNCCC=C)cc1 C1(C(=O)N(CCO)CCCC)(OC2CC2)CCOCC1.C(=O)(COC(C)CC)N C1(C#N)(COC)CN(C(=O)CC2CCC(NC(=O)C(C)OC)C2)C1 CC1(CNC(C2(C)CCCOC2)=O)CCN(C(c2ccc(CO)s2)=O)CC1 CCCCC(C)CCC(=O)N(CCN(C(C1CCC(N(C)C)CC1)=O)CC)CC N1(C(CCc2ccn(C)c2)=O)CC2C(CNC(c3ccc(CF)cc3)=O)C2C1 N1(C(CSCCC(C)C)=O)CCC(C)C(CNC(c2cc(C#N)n(C)n2)=O)C1 C1(C(=O)NCCN(C(CN2CC(=O)NCC2)=O)CC2CC2)CC2COCC2C1 N1(C(CN(C(C)C)C(c2ccc(=O)oc2)=O)=O)CCOC(C)C1 C(=O)(CCCC(N)=O)NCCCNC(C(N1CCCC(O)C1)C)=O C12(NC(CCC=C)=O)CCC1CN(C(c1cc(-c3cccc(Cl)c3)no1)=O)C2 C(F)(C(=O)N(C)CCOCCCNC(=O)Cc1cnoc1)OC c1(NCc2c(OC)cccc2)ccc(N2CCOCC2)cc1Cc1ccccc1 C1(C)(NC(CCNC(COC)=O)=O)CCCCC1C(N1CCCCC1C)=O N1(C(c2scc(C#N)c2)=O)CC2OCC(NC(=O)CCn3cncn3)C2C1 c1(OC)ccc2c(ccn2CC(N2CCC(NC(=O)C=CS(C)=O)CC2)=O)c1 O=C1CC(C(=O)NC2(CNC(=O)C(F)(F)c3cnccn3)CCCC2)CCN1 C1(C(N(CCCCN(C)C(C2(c3cccc(Cl)c3)CC2)=O)C)=O)CC(C2CC2)C1 C1(NC(C2C(OC)C2)=O)CN(C(c2coc(OCC(F)(F)F)n2)=O)CC1(C)C C1(C(N2CC(F)(C(=O)NCC3(F)CC(CO)C3)C2)=O)CCNC1=O N1(C(C(CC)SC)=O)CCCC(NC(c2ccc(OC(C)C)nc2)=O)C1 C1(NC(=O)CSc2ccncc2)CC2CN(C(=O)CCc3ccncc3)CC2C1 CC(CBr)C(=O)N1CCCC1Cc1cn(Cc2cnoc2C2CC2)nn1 C#Cc1ccc(C(=O)NC2(CC=C)CN(C(=O)C(CC=C)CC=C)C2)cc1F Cc1cc(C)n(CC(N2CCC(C(C)C(N3CCC(CN=[N+]=[N-])C3)=O)CC2)=O)n1 c1(NC(C(CN(CCN(C)C)CC)CC2CC2(C)C)=O)cnc(Cl)c(C)c1 c1(SC)ccc(Cl)c(C(N2CCC(N(C(=O)Cc3nncn3C)CCO)C2)=O)c1 c1(NCC2(O)CN(C(c3c(OC)noc3C)=O)C2)ccc([N+](=O)[O-])cc1C CCCCC(=O)C(=O)NCCCCNC(C1CCCC(C2CC2)O1)=O N1(C(C2C(C(=O)OC)C2(C)C)=O)CC2CC2(NC(=O)Cc2scnc2C)C1 c1(C(=O)NC2CN(C(C(CC=C)(C)CC)=O)C2)cc(Cl)c2c(c1)OCO2 C(C(CC(C)C)C(=O)N(C(C)C(=O)OCCOC)C)c1c(OC)c(F)ccc1 CC1=C(C(=O)NC2CCOC(C(=O)NCc3cc(=O)cc[nH]3)C2)SCCO1 c1(C(=O)NCCNC(c2nn(C)c3c2CCC3)=O)ccc2c(c1)CCC2(F)F CCCC(C)C(=O)NC1CN(C(c2cnn(CC)c2C)=O)CC1c1ccccc1 N1(c2nc(C)nc(Cl)c2)CC(NC(C2OC(C)CC2C)=O)C2(CCOCC2)C1 c1(C(=O)NC(C2CCCN2C(C2CC(=O)N(O)C2)=O)(C)C)cn2ncccc2n1 N1(C(C)=O)CCC(N=c2[nH]c(C(C)(C)C)no2)C1 C1(NC(Cc2c(C)noc2C)=O)CN(N(c2ccncc2N)C)CCC1C C1(CNC(CCCC(C)C)=O)CCC2CN(C(=O)CC(C)N(C)C)CC12 c1(C2C(C(=O)NCc3ccccc3CC(F)(F)F)CC2)cccc(F)c1 c1(C(C)=O)cc(C(=O)NC2CCC2NC(C2(C3CC3)CC2)=O)ccc1Br N1(C(c2cc(OC)no2)=O)CCCC(NC(C2CCC(=O)N2C)=O)CC1 C(C(CNC(c1cc(C2CC2)nn1C(C)C)=O)C(C)C)OC c1(C(N(C)CCNC(=O)C(=Cc2cccc(F)c2)F)=O)cnc2occc2c1 c1(C(=O)OC)cc2c(N(CC(C)NC(=O)CC3CC(C)(C)CO3)C)[nH]cnc-2n1 C(=O)(C(F)CC(C)(C)NC(=O)C(CO)C(F)(F)F)NCC(CC)CC(C)C C1(C(c2nnnn2C)NC2C(c3cn(C(C)C)nc3)OCC2)(CCl)CCOCC1 N1(C(c2ccc(OC)nc2)=O)C2CCCC1CC(NC(=O)C=C1CCOCC1)C2 C1(CC)CN(C)C(=O)CN1C(=O)CCCCCN(C)C(C1CC(=O)N(OC)C1)=O CCS(=O)CC(=O)NCCCN(C(c1cccc(-c2noc(C)n2)c1)=O)C1CC1 C1(C)(C(N(CC)CC)=O)CC12CCN(c1nccc(N)c1OC)CC2 Cn1ncc(C(=O)NC2CCCC2(C)C)c1F N1(C(CCCN(C(C)=O)C)=O)CCC(C)C(CNC(=O)CNc2cnn(C)c2)C1 c1(-n2cnc(NC(C(CC)O)=O)n2)ccc(NS(=O)(=O)CC)cc1 c1(CC)c(C(=O)N(CCC(C)NC(=O)C(C(C)C)c2cnn(C)c2)C)csc1C C1(NC(CCC#C)=O)CC2(C1)CC2C(=O)NCc1cncc(C)c1 c1(OC)ccc(C)cc1C(=O)NCC1CC(NC(=O)C=C2CN3CCC2CC3)C1 c1(OC)ccc(C(N2CCCC2CC(=O)NCC2C3CCCOC23)=O)nn1 CN1CCOc2ccc(C(N3CCC(CCNC(=O)C(F)=C4CCC4)C3)=O)cc21 C1(CNC(CCCC)=O)CCN(C(c2nnn(C(C)C)c2C)=O)C(C)C1 Cc1[nH]c(C)c(NC(C2CCN(C(=O)COc3cccc(C(=O)O)c3)C2)=O)c1C Cc1cc(C)n2nc(C(=O)NC3(C)CCC(NC(C45CCC4C5)=O)CC3)nc2n1 N1(C(C(CC)C)=O)CCC2(CC1)CC2NC(c1cc(F)ccc1C)=O C=C(Br)CCC(=O)NCC(C1CCN(C(=O)C(C)n2ccnn2)CC1)F C1(NC(C(CCOC)NC(=O)CCC2OCCO2)=O)CCc2nncn2C1 N1(C(C2CCC(C)O2)=O)CCC(C2CC2)(CNC(=O)CCn2ncn(C)c2=O)C1 C1(C(=O)NCC(c2ccccc2)F)COCCN(C(c2c[nH]cc2C2CC2)=O)C1 c1(CCNC(c2nc(C)nn2C)c2nnnn2C2CC2)c[nH]c2cccc(F)c12 N1(C(C(C)SC)=O)CCCC(NC(=O)CN(CC(=O)NCCOC(C)C)C)C1 CC1CN(C(=O)CCOCCN(C)C)CC1CC(=O)N(C)CCn1cccn1 C1(CC=C)(C(=O)NCC2(n3nccn3)CC2)CCCN1C(=O)CC1CC2CC2C1 c1(C(N2CC3(CCC(C(=O)NCC(C)(C)C)O3)C2)=O)cc2ccc(Br)cc2s1 CC1(C)OCCC1CC(=O)NCC1CC(NC(=O)CNC(=O)C2CC2)CC1O N1(C(c2ccc(Cn3cc(CCCCCO)nn3)o2)=O)CC2CC3CC2C1C3 N1(C(c2cn(CCCC)nn2)=O)CC(NC(=O)C(CC)SC)C2CC2C1 Cc1noc(C(C)C)c1NC(=O)CC1CN(C(c2cnn(CCO)c2)=O)CC1C Nc1nn2ccccc2c1C(=O)NCCC1CCN(C(=O)C=CC2CCC2)CC1 Cc1ccc2occ(C(N3CCC4CCN(C(=O)C=CCF)CC34)=O)c2c1 c1(OC)ccc(F)cc1C(N1CCCC(N(C(=O)COCC(F)F)C)C1)=O c1(NC(C(N2CCC(C(=O)NCCC)C2)=O)=O)c(OCC)ccc2c1CCC2 C1(C(=O)NCC2(C)CCCCC2O)(COC)CCN(C(=O)CC2CCCC2)CC1 N1(C(CCN(C)C)=O)CCCC1CC(N1CC(C)(CN(C)C)C1)=O c1(C(=O)NCCC(C)NC(CCc2cnc(C)o2)=O)cnc(Br)c(N)n1 Cc1ccc(CCC(=O)NC(C(=O)NCCOCCCO)C2(O)CCC2)o1 N1(C(C2N(C)CC2)=O)CC2CC(C1)CN(C(C1(C)CCCO1)=O)C2 c1(COC)cccc2[nH]c(=NC(CO)C(C)C)sc12 C=CC1(C(=O)OC)CCN(CCCCO)C1 N1(C(C(CSC)O)=O)CC2(CNC(=O)CCc3nccn3C)CC1CCO2 c1(C(N2CC(C)CC(NC(C(CC)(C)O)=O)C2)=O)ccc(F)c2c1CCC2 C1(NC(C(C(C)C)OCC)=O)CCC2(CCN(C(=O)Cc3ccco3)C2)C1 C1(C(=O)NC2CC(CNC(=O)CC(C)c3cccnc3)C2)(OC)CCCCC1 C#Cc1ccc(C(=O)NCCC2CC(OC)CN2C(=O)COC(C)=O)cc1C Cc1ccc(Cl)c(O)c1C(N1CC2(COC(CNC(c3coc(Br)n3)=O)C2)C1)=O c1(C(=O)NC(C)CCN(C)C(C2COC(=O)O2)=O)cnc2n(c1=O)CCS2 c1(NC2(C3CN(C(C(C)(C)N4CCCCC4)=O)C3)CC2)ncc2c(n1)CCOC2 c1(C(=O)NCC(CCNC(=O)CCCn2cncn2)OC)cccc(F)c1 c1(CC)cnc(C)c(NC(=O)C(C)=CCNC(=O)COC2CCC2)c1 C1(C(=O)NC2(C=C)CCCCC2)CC(C)(C)OC1(C)C.C12CN(CC1C)C(=O)C2 Cc1cc(NC(=O)C(C)C(=O)O)ccc1-n1cncn1 CC(C)(C)C(C)(C)C(=O)NCC1CCN(C(C2CN(S(N)(=O)=O)C2)=O)C1 N1(C(Cn2c(C)cc(C)n2)=O)CC(NC(c2cc(C)n(C)n2)=O)CC12CCCC2 C1(C(N(C(CNC(Cc2nc(CC)sc2)=O)C)C)=O)CC(C)(C)CCO1 CCCC(CCNC(=O)C1=NOC(CNC(C2CC=C(C)CC2)=O)C1)CCC S(=O)(=O)(c1c[nH]ccc1=NCC1CCCOC1)NC(c1ccc(Cl)cc1)C C1(CNC(C(=O)NC(C2CCCC2O)C)=O)CCN(c2ccccc2)C1 C1(CC(=O)NC2CCN(C(=O)CC3(C)CC3(F)Cl)CC2)(CN(C)C)CCOCC1 Cc1oc(CNC(=O)CC2CNC(=O)O2)nc1C(N1CCCC1(C)C(C)(C)C)=O N1(C(C2(OC)CCCC2)=O)CCC(C)C(CNC(C2(F)CCCC2)=O)C1 C1(OCCC)CCCN(C(=O)NCCCCCCN(C)C)C1 c1(OC)cc(OC)c(C(N2CCN(C(=O)Cc3ccsc3)C(C(F)F)C2)=O)cn1 c1(OC)ccc(CNC(N2CC3(NC(=O)C=CC(F)(F)F)CCC2C3)=O)c(C)c1 C=CC(CCC)CC(=O)N1CCC(C)(NC(=O)CC2C=CCC2)CC1 C(=O)(CCC(=O)N1CCC(C(C)C(=O)NCC(C)(CC)OC)C1)OCC C1(C(=O)NCC(CC)(CC)NC(=O)C#CC(C)(C)O)CCc2cncn2C1 c1(COCCOC)ccc(C(=O)N(CC(C)NC(C2(C)C=CCC2)=O)C)cc1 C(CC(=O)Nn1ccnn1)(C(C)(C)C)NC(c1c(C)cc(C)s1)=O c1(NC(C2CCCOC2)CC)cc(-c2cccs2)ncn1 c1(C(=O)NC(C)C)cccc(NC(=O)NCCC(O)C(=O)O)c1 C(CCCC(=O)NCC1CCCN(C(=O)C(c2ccccc2)O)C1)N(C(C)=O)C N1(C(c2c(C)ccc(C)n2)=O)CCN(C(=O)Cn2cnnn2)C(C)C1C N12CC3CN(C3C1)C2.c1ccc(C(F)(F)F)nc1.CC1(C=O)CCCC1 c1(C(n2cc(CN(C3CCN(N(C)C)C3)C)nn2)O)ccccc1Br CC1CCC=C1C(=O)N1CC(NC(c2ccc(OCF)cc2)=O)C2(CC2)C1 Cc1cc(C(N2CCC(C)N(C(c3nnsc3N)=O)CC2)=O)c(C)c(C)c1 N1(CCC(=O)NCC(CNC(c2c(CC)nccn2)=O)(C)O)CCP(C)(=O)CC1 c1(CC)cc(C(N2CCOCC(NC(c3csc4cncn34)=O)C2)=O)cc(O)n1 N1(C(C23CCC(OC)C2C3)=O)CCC(C(=O)NC(C(C)C)C2CC2)CC1C C1(C2CCN(C(C3(CC=C)CCC3)=O)C2)CCCCN1C(=O)CN1CCOCC1 c1(CCNC(C=CC(C)NC(=O)C=CC(C)(C)C)=O)noc(=O)n1C c1(CN2CC(F)(C(=O)Nc3cc(O)nc(O)n3)C2)c(F)c(F)cc(F)c1F c1(N2C(=O)CCN(CCC(CC)C)C2=O)ccc2c(c1)OCCCO2 C(=O)(CCCC(=O)NCC)N1CC(CNC(COCC(=C)C)=O)C(C)C1 c1(C(N2CC(C)C(CNC(=O)C(O)C(C)(C)C)C2)=O)cc(F)c(CO)c(F)c1 c1(C(=O)NCC(CNC(C2(OC)CCCOC2)=O)O)cc2ccccc2nc1O Cc1nc(C(N2CCC2Cn2cc(CCC#N)nn2)=O)ccc1N1CCOCC1 N#Cc1c[nH]c2ccc(C(N3CC4CC(NC(c5csnn5)=O)CC3C4)=O)cc12 C(=O)(C(CC(C)C)C(N)=O)N1CCC(C(=O)NCC2C(OC)CC2)(CC)CC1 C1(NC(=O)Cc2ccn(C(F)(F)F)n2)(CF)CCN(C(=O)CC2CSC2)C1 N1(C(c2ccc(CC)o2)=O)CC(NC(C2CCCN(C)C2)=O)CCC1C N1(C(c2c(CC=C)cccc2)=O)CC(C)(C)CC1CNC(C1CCCOC1)=O C(=O)(CC(C)(C)C(=O)NCC(C1CC1)N(C(=O)CNc1ccccn1)C)OCC C12(C(=O)O)CCCC1(C(N1CCCC1Cc1ccc(Br)cc1)=O)C2 C=CCC(CNC(C1CSCCN1C(=O)C=C(C1CC1)C1CC1)=O)CC(C)C c1(C(=O)OC)ccc(Cl)c(CNc2cccnc2C(=O)Nc2nn[nH]n2)c1 Cc1ccc(CC(N2CC3C(C(=O)N(CC(C)C)C)C3C2)=O)cc1 c1(C(N2C(CNC(C=CC(=O)N(C)C)=O)CCC2)=O)cc(=NS(C)(=O)=O)cc[nH]1 c1ccnc(Br)c1F.C1(C)(OC(C)=O)CCC1.C12CC1C(=O)N(CC)C2=O n1(CC=C)nnnc1C(c1ccn(C)n1)NCC1(CCO)CC1 C(C(C)C(=O)N1CC(CNC(=O)Cc2ccc(C(C)=O)s2)C1)OCC c1(C(=O)NC2(CNC(c3cc(Cl)c[nH]3)=O)CC3CCC2C3)ccnc2ncnn12 n1(C(C)C(=O)O)cc(CN(CCCO)Cc2ncn(C)n2)nn1 C1(CNC(C2(CC#C)CC=CCC2)=O)(CO)CCN(C(C2CC2F)=O)CC1 Cn1cnc(C(=O)NCCN2CCCN(C(=O)CC3=CCCC3)CC2)cc1=O c1(CC(N2CC(NC(C3N(C)CCCC3)=O)CC2(C)C)=O)c[nH]c2cccnc12 Cc1cc(C(=O)NC2CC2NC(c2cnoc2-c2cccs2)=O)on1 CC1OCCCC1C(=O)N(C)CCOCCN(C(=O)Cc1cccnc1)C C(C1=CCCCC1)NC(CC1N(C(CC=CCCCCC)=O)CC1)=O c1(C(N(C(C(=O)OC)C)C)=O)ccc(CNC(C2(C3CC3)CCCO2)=O)s1 N1(C(C(=O)NCCCSC)C2CCOC2)CCCC2(CCCC2)C1 C(C(CCC)CCC)NC(C1C(NC(CCOCC#C)=O)CC1)=O C=CCCCC(C(=O)NC(c1nc[nH]n1)C)NC(c1ccc(C=C)cc1)=O CC(F)(F)C(=O)NC1(CO)CN(C(=O)CN2CCCC2CO)C1 c1(C(=O)NC2(C)CCN(C(c3ncsc3C3CC3)=O)C2)cc2ccccc2[nH]1 C(=O)(C(F)CCCC)NCC(CCCC)NC(c1cc(C)oc1CC)=O C(=O)(CCC(CC)CCC)NC(CC#CC)C(=O)N(CC(O)COC)C c1(C(N2CCOC(COC)C2)C(=O)NCCC(=O)OCC)cncc2ccccc12 C#CCC(CC(F)F)C(=O)NCCOCCNC(c1ccc(C(C)=O)c(O)c1)=O C(=O)(C(C)(C(C)C)OC)N(CC1CCN(C(C2C(C#C)C2)=O)CC1)CC c1(OCC=C)ccccc1C(=O)N(c1nnc(Br)n1C)CC C(=O)(C(CC(C)C)N(C)C(c1coc(C)c1)=O)N1CCC(OCC=C)CC1 c1(CC#C)ccc(C(=O)NC2CC(N(C(=O)CCC=CCC=C)C)C2)cc1Br c1(NC(C)=O)cccnc1C(=O)NCC(C)NC(=O)C(c1ccc(F)cc1)(C)F C(=O)(CC1=CCOCC1)N1C(C(=O)NCCC(O)CO)CC(O)C1 C1(CCNC(C2CC(=C)C2)=O)CN(C(c2ccc(-c3cnco3)cc2)=O)CCO1 CN=c1ccc(C(=O)N(C)CC2CCCN2C(=O)CSC(C)C)c[nH]1 CN1CCC(NC(=O)C2=CCCO2)C12CCCN(C(=O)C(C)(C)C(C)(F)F)C2 C1(NCc2ccc(OCCN(C)C)cc2)CC2CCC(C1)N2C C(=O)(CCCCCC#N)NC(C(=O)NC1C(SC)CCC1)CCSN(C)C C1(CNC(c2cc(C)c(Cl)s2)=O)CCC(C)CN1C(c1cn2ccnc2s1)=O c1(C(N(CC(C)NC(CCCC(=O)OCC)=O)C)=O)ccc2c(c1)COCC2 C1(C(N2CCC(C(C)NC(=O)CCC3CCCOC3)CC2)=O)C2C3CCC(C3)C12 C(CC(C)(C)CC(=O)NCCC(C)NC(c1cnn(C2CCC2)c1C)=O)OC c1(CC)sc(=N)[nH]c1C(=O)NCC(C)(O)CNC(=O)Cc1cnccc1Cl c1(CNCC(Cc2ccccc2)N(C(=O)CCF)C)ccc(F)c2cnccc12 N1(C(C2(C#N)CC3CC3C2)=O)CCOC2(CCN(C(C3CC(=O)N3)=O)C2)C1 n1(CC)nccc1C=CC(N1CC(NC(c2cc(C)c[nH]2)=O)CC1CO)=O C=Cc1cc(C(=O)NCC(C)CNC(c2cccc(F)c2C)=O)cc(F)c1 N1(C(CC(C)N(C)C)=O)CCC(O)(C2CCN(C(C3CC3C(F)F)=O)CC2)CC1 CCCCC(C)(F)C(=O)N1CCN(C(C2CC2(Cl)Cl)=O)C(C)C1 C1(COC)(NC(=O)CCCn2cccn2)CCN(C(=O)CC2C(=O)NN=C2C)C1 C1(NC(c2cncc(CC)c2)=O)CC(O)CN(C(c2ccc(CO)cc2)=O)C1 CCC(C)(C)CC(=O)NCC1(O)CC(NC(=O)CCCc2ccsc2)C1 c1(CCC(=O)NC23CC(CNC(C(CC)NC(N)=O)=O)(C2)C3)ccc(Cl)c(C)c1 c1(C(=O)NCCNC(COc2cc(C)c(Cl)cc2)=O)ccc2c(c1)C(=O)NCC2 c1(CN2CC(C)N(C(C3CCCS3)=O)CC2)ccc(O)c([N+](=O)[O-])c1 Cc1cc(C(N2CCN(C(=O)Cc3cc(C4CC4)no3)C(CO)C2)=O)ccc1F c1(SC)ncc(C(=O)NC2CC3CC2N(C(=O)C(C)NC(C)=O)C3)c(O)n1 NS(=O)(=O)CCCC(=O)NC1COCCN(C(C2CC2C2CCCC2)=O)C1 c1(OC)cc(C(=O)Nc2ccc(C)c(C)c2)cc(Br)c1OC c1(NC(C2(F)CCCN(C(CSCC)=O)C2)=O)c(F)cc([N+](=O)[O-])cc1Br C#CCC(CC(=O)OC)NC(C1CCCN(C(C2(OC)CC2)=O)C1C)=O N1(C(c2nc(C(C)C)sc2)=O)CCC2OCCN(C(=O)C#CC3CC3)C2C1 CC1CCN(C(c2cc(F)cc(Cl)c2)=O)C(CNC(=O)CNc2ncccn2)C1 C=CCCCC(N)C(=O)N1CCCC(O)(CO)CC1 N1(C(C2(C#N)C(C)(C)C2)=O)CCN(C(C2CCCCC(F)(F)C2)=O)C2(CCC2)C1 C1(C)(CC)CCCN(C(c2ccc(CNC(=O)C(C(=O)OCC)OC)nc2)=O)C1 C1(C(N(CCN(C(c2ncc(Br)cn2)=O)CC)CC)=O)CCCC(C#N)C1 C1(CCC)CCC(O)(C(=O)NCCCC(C)(C)NC(=O)C(O)C(F)(F)F)CC1 C#CCC(C(=O)NC)NC(c1cc(CNC(C2C=CCC2)=O)ccn1)=O c1(CN(CCCN(CC(CCCCC)CC)C)C)cc(=O)oc2cc(C)ccc12 C(CCC(CCC)NC(=O)CC12CC(C1)C2)NC(C(C)SCCCC)=O c1(C(N2CCCC(C3N(C(COCC)=O)CCC3)C2)=O)cc2cc(Cl)ccc2[nH]1 c1(C(C(=O)NCC(C)N(C(C2COC(=O)N2)=O)CC)(F)F)ncccc1F N1(C(C2C(CC)OCC2)=O)CCC2CN(C(c3cnccn3)=O)CC12 N1(C(c2c(C)c(Br)cs2)=O)CCCC(O)(CNC(c2cncn2C)=O)C1 CC(O)(C(=O)NCCCCNC(=O)CCC1CCCC1)c1ccccn1 c1(OCC(C)C)cc(C(=O)N(CCN(C)Cc2ccc[nH]2)C(C)C)ccn1 c1(NC(CC)CNC(C2(C)CCOCC2)=O)ncnc2sc3ccccc3c12 c1(C(=O)NC(C)CN(C)C(C2(n3cnnn3)CCOCC2)=O)cnc(O)cc1O C(=O)(C(O)CNC(C1CC(C)(F)C1)=O)N(C)Cc1cncs1 c1(C(=O)NCC2N(C(c3ccn(CC)c3C)=O)CCCC2)ccc2c(c1)OCO2 C1(COC(c2cccn2C(F)F)=O)CCC(Cc2ccncc2)C1 CCC(CCOC)C(=O)N1CC2CC2C1C(=O)CCNc1cccc(OC)c1 c1(C(C(=O)NCCOC)N(CCCO)C(C)C)nccc(Cl)c1Cl C12(CN(C3CC4CNC3C4)C(c3cnn(C)c3Cl)=O)CC1COC2(C)C C(=O)(C(C)CC(C)(F)F)NC1CCN(C(c2c(CC)ocn2)=O)C12CC2 c1(Cc2c(OC)cccc2)nc2ccc(=NC(CSC)CO)[nH]n2c1Br Cc1ccnc(C)c1C(=O)NCC(C)CNC(=O)CCn1ncn(C)c1=O C(=O)(C(C(C)(C)C)N1CCCC1=O)NC1C(NC(c2c(C(C)=O)nccc2)=O)C1 c1(C(=O)NC2C3CCCC2CC3)ccc2c(c1)CN(C(=O)Nc1ccccn1)C2 c1(N(C)C)nc(C(N2CC3(NC(=O)CCC4CC4(F)F)CCC2C3)=O)cc(O)n1 C1(NC(Cc2c(C)n[nH]c2C)=O)CC(C)CN(C(c2ccc(CO)nc2)=O)C1 CC(CCCCNC(=O)C(N)=O)NC(=O)CCC(=O)NC1CCCC1 CC1CC(C(=O)NCc2cn(C3CN(C(=O)CSC(F)F)C3)nn2)CO1 C(O)(CN=c1cccc(S(=O)(=O)NCC2C=CCC2)[nH]1)c1ncn(C)c1 CCC(C)(C)C(=O)NCc1ncccc1NC(=O)C(CNC(=O)OC(C)(C)C)OC C1(CNC(CSc2c(C)n[nH]c2C)=O)CC(F)(F)CN1C(c1ncn(C)c1C)=O N1(C(c2n(CC#C)ccc2)=O)CCC(C)(C)C(C(=O)NCC(C)CC(C)C)C1 C1(C(N2CC(NC(C3COCCO3)=O)C2)=O)CCCN1Cc1cccnc1 Cc1cnn(C)c1CC(=O)NC(C)(CNC(=O)Cc1cnn(C)c1)CO N1(C(C(=O)NCC(C)C(=O)O)=O)CCCC(OCc2cn(C3CCCC3)nn2)C1 C(C(C)(C(=O)NC1CC(NC(c2snnc2C2CCC2)=O)C1)OC)OC Cc1nn(C)cc1C1=NOC(C(N2CCCC2C(C)NC(=O)C=C(Cl)Cl)=O)C1 c1(C(N2CC(NC(C(COCC)C)=O)C3C(C2)C3)=O)noc2c1CCCC2 C1(CC)CN(C(C2COC3(CCC3)C2)=O)CCN1C(=O)CSC(C)(C)C C=CCC(C)(C)CC(=O)N1CC=CC1CNC(=O)CCC(C)OC CC(CC(C)(C)C)C(=O)NCCC1CCN(C(=O)C(F)(F)CN(C)C)C1 c1(C(N2CC(CNC(CCCOCC=C)=O)C(O)C2)=O)coc2ccc(F)cc12 C1(NC(=O)CC2CC3CCC2CC3)CC2CC1CN(C(=O)Cc1cnoc1)C2 c1(SC)nc(C(=O)NCC2CCN2C(=O)CCc2cnc(C)s2)c(C)c(Cl)n1 N1(C(C(C)OCCC#C)=O)CCC(N(CCC)C(c2cc(C(C)(C)C)on2)=O)C1 CC1CN(C(=O)CC(F)F)CC1NC(c1cc(N2CCC(O)CC2)ccn1)=O c1(C(N2CCC(N3CC(C)(C(F)(F)F)C3=O)CC2)=O)cc2ccc(F)cc2s1 C(=O)(CC(C)C(F)F)N(CCC(=O)NC(C)CCN(C)C)CCCO c1(CCNC(C(C)OC(c2cc(C(F)(F)F)n[nH]2)=O)=O)ccccc1 Cc1ccc(OCC(N2CCC(CNC(C3CC4CC4C3)=O)C(C)C2)=O)cc1C C1(NC(c2coc(C(F)F)n2)=O)C2CC1N(C(=O)Cc1cccnc1Cl)C2 C(CC(=O)NC1(c2ncc(C)o2)CC1)(C(F)(F)F)NC(c1nc(COC)oc1)=O c1(C(=O)NC2CN(C(C3C(C=C)C3)=O)CC2C)cc2cnn(C(C)C)c2nc1C C(=O)(C(CCc1ccccc1)OC(=O)COCC1CCC1)OCC c1(CC)cccc(CN2CC(C(C)NC(c3cnc(CC)s3)=O)C2)c1 N1(C(C(c2ccnn2C)C)=O)CCOCC(CNC(c2cncc(F)c2Cl)=O)C1 Cc1cc(C(=O)NC2CCC(CNC(=O)C(C)NC(N)=O)CC2)ncn1 c1(CCC(=O)N(C2CCN(C(c3nocc3C)=O)C2)CC#C)ccc(C)c(C)c1 C1(C)(C(=O)Nc2cnc(CCC)nc2)CN(C(C2CC(CC3CC3)C2)=O)C(C)(C)C1 Cc1cc(N(CC2CC(C)CN2C(=O)C#CC(=O)O)Cc2ccccc2)nc(C)n1 Cc1nn(CC(=O)NCC2CCN2C(C2CC3CC3CC2C)=O)c(=O)n1C C(C(N=[N+]=[N-])C(=O)NC(C(N1CCC(F)(C#N)C1)=O)C1CC1)OCC N1(C(C=CCC)=O)CCC2(CCCCN(C(=O)Cc3csc(C)n3)C2)C1 C(=O)(N=c1[nH]n(CC2CC2)cc1C#N)C1CCC(CNC(=O)OC(C)(C)C)CC1 c1(-c2cnc(CCN(CC(C)C)C)nc2)ccccc1C#N c1(C(=O)NCCC(C)N(C)C(c2cccc(F)c2Cl)=O)cccc2c1CCO2 C12(CN3CCCC(COC(C)=O)C3)CNCC1COC2 N1(C(C(C)=O)=O)CCC2(CCC2NC(C2CCNC(=O)C2)=O)CC1 c1(OCC)cc(Br)ccc1C(N1CC=CC1C(N1CC(O)C(F)C1)=O)=O Cc1cc(C(N2CCCC2CCCNC(=O)C(C(C)C)NC(N)=O)=O)c(C)s1 c1(C(C)C(=O)Nc2cccc(F)c2)cccc(S(=O)(=O)N2CCN(C)CC2)c1 C12(CNC(C(C)OC)=O)CC1CN(C(=O)COC1CCCOC1)C2 CCCCCC(O)CC(=O)N(CCN(C(=O)CC(CC)C(F)F)C)C(C)C c1(-c2nc(CCCSC)nn2C2CCC(C)C2)ccc(F)c(COC)c1 CC(C)C(CN(C)C)C(=O)NC1CCN(C(=O)C(N)=O)CC1O C1(C(=O)NCCC2(C(N(CC(O)CO)CC)=O)CC2)CCCCS1 Cc1cc(F)cc(Cl)c1NC(=O)CC1CCN(C(=O)Cc2cccc(Cl)n2)CC1 N1(C(C(C2CC2)SC)=O)CCC2C(C1)CN2C(=O)Cc1nocc1C C1(C(N2CCC2c2cn(C3CCCC=C3Br)nn2)=O)CN(C2CC2)CC2(CCC2)C1 N1(C(C(=O)N(C)CC2CCCSC2)=O)CCOc2ccc(Cl)cc2C1 Cc1nnc2c(C(=O)NCC3(F)CC(CNC(=O)Cc4cnoc4)C3)cccn12 Cc1ccc(CN(C=O)Cc2ccc(O)c(Cl)c2)cc1C(F)(F)F N1(CC(=O)N(CC(C)NC(=O)C(C)n2ccnc2)CC)CCP(C)(=O)CC1 C#CCC(CC#C)C(=O)NC1CN(C(C2(C)CCC2)=O)CC1c1ccc(F)cc1 N1(C(C(C)OCC)=O)CC2(C1)OC1(C)CC2(NC(C2COCCN2C)=O)C1 S(=O)(=O)(c1ccc(=NCC2CC2)[nH]c1)NC(c1cc(C)cc(C)c1)CC c1(C(C)C)cc(CC(=O)N(CCC(C)NC(=O)CCc2cnn(C)n2)C)on1 N1(C(c2cc(C)sc2)=O)C2CCC1CC(C(=O)Nc1cnn(C)c1C)C2 C(=O)(C(CNC(=O)C1=CCC(C)CC1)(CC)CC)N(CC#C)C c1(C(=O)NCC2(OC)CN(C(C3CN4CCN3CC4)=O)C2)c(F)cc(F)cc1Cl c1(C(C)NC(=O)C(N)=O)ccc(SCCNC(=O)C(F)(F)CN(C)C)cc1 Cc1c(Br)cc(Cl)c(NC(=O)CC2CCCN2C(c2ncccn2)=O)c1Cl C1(C(=O)NCCCNC(C2(c3ccn(C)c3)CC2)=O)CCC(C(F)(F)F)CC1 C1(C(=O)NC2COCCC2NC(C23CCC(CC2)C3)=O)CC2CCCC(C1)C2 C1(CNC(c2c(COC)scc2)=O)CCCCN1C(C1C(C(F)F)C1(C)C)=O N1(C(c2c(C(C)C)onc2)=O)CCCN(C(=O)CCSCC2CCCO2)CCC1 c1(C(C)=O)cnccc1C(=O)NCC(F)CNC(C1OCCOC1C)=O N1(C(c2c(CC)con2)=O)CCCC(C(N2CCC23CCC3)=O)C1C Cc1cc(C(N2CC(O)CC2(C)C(=O)NC2(c3ccsc3)CC2)=O)nc(O)n1 N1(CC(=O)NC2(C)CC(NC(CC(C)O)=O)C2)C(=O)NC2(CCOCC2)C1=O c1(SC)csc(C(N2CC(OCCNC(=O)CC(=O)NC3CC3)C2)=O)c1 N1(c2ccc(F)cc2)CCC(N=c2nc(N3CC4CCC4C3)c3sccc3[nH]2)C1 CCS(=O)(=O)CC(=O)N1CCCC1(C(=O)NC1CC2(CCC2)C1)CC N1(C(CCCNC(CCSCCCC)=O)=O)CCC(C)C1(C)C C1(C(=O)NC(CN(C(C)C)C)C)CC(=O)CN1C(c1ncc[nH]1)=O N1(C(C(C)(Cl)CCl)=O)CC2(CC(C(=O)NC3CC3(F)F)CO2)C1 N(C(=NCCF)NC1CCN(C2CC2)CC1)Cc1cccc(C(C)O)c1 Cc1cc(C(=O)NCC#CCNC(=O)Cn2cnc(C(N)=O)n2)nc(O)c1 C1(NCc2ccc(C)cc2)CCN(S(=O)(=O)c2ccccn2)CCC1C N1(C(C(N2CCOCC2)C)=O)CC2CCCC2(Nc2nccc(C(C)(C)C)n2)C1 Cc1cc(C(N2CCCN(C(=O)C(C)NC(N)=O)CC2C(C)C)=O)c(O)nc1C CC1(C)CN2CCN1N1CCC(F)(C1)C2=O.c1(C[SH](=O)=O)c(F)cccc1F.CCN N1(C(c2ccc(CC)o2)=O)CCC(CCOC)(NC(C2COC(=O)N2C)=O)C1 c1(C2(C(N(CCNC(COC(CC)C)=O)C)=O)CC2)ccc2c(c1)OCO2 c1(OC)cc(N(CCCNC(C2CCCC(C)C2)=O)C)c(F)cc1[N+](=O)[O-] C1(C(N(CC(O)CNC(c2csc(-c3cn[nH]c3)c2)=O)C)=O)CCCCS1(=O)=O CC1CCCN(C(=O)COC(c2cc(C3CCOCC3)nn2C)=O)CC1 N1(C(CNC(C(CC)C)=O)=O)Cc2nccn2CC(NC(c2ccc(Cl)[nH]2)=O)C1 C1(CC=C)(C(=O)NCCC2CCC(NC(C3OCCO3)=O)C2)CCCCC1 c1(CC)cccc(C(=O)NC2CCC(NC(=O)C(C)(C(C)C)OC)CC2)c1N C(=O)(C1=Cc2ccccc2OC1)N1CC(N(C(=O)C(Cl)=CCl)C)C(C)(C)C1 C1(NC(C2(C#C)CCC2)=O)CCN(C(c2cccnc2S)=O)CC1CC c1(CC(N2CC(CNC(C=Cc3nnn(C)n3)=O)C2)=O)cc(C(F)(F)F)cc(Cl)n1 c1(OC)cc(F)c(C(N2CCC(NC(c3cncc(F)n3)=O)C2)=O)cc1OC N1(C(C(C)=C(CC)C)=O)CCOC(C(=O)NCC(C)(C)C(C)O)C1 N1(C(CNC=O)=O)CC2CC2(CNC(C2CCC2c2nc[nH]n2)=O)C1 C1(C2CC2)(CNC(=O)CCC2CCCO2)CCN(C(c2cnc(C(F)F)s2)=O)C1 c1(C(=O)NCC2(F)CC(NC(C(C)(C)O)=O)C2)nccn2c(Br)cnc12 N1(C(c2c(CC)noc2)=O)CC(F)(F)CC1CNC(=O)Cc1occc1C c1(C(=O)OC)c[nH]c(=NCC2CN(C(C3COCCO3)=O)CC2C)cc1[N+](=O)[O-] C(=O)(C1CCc2c[nH]nc21)NCC1CCCCN(c2nc(C)cc(SC)n2)C1 CCC(O)C(C)C(=O)NC1CC(F)(CNC(c2cnn3ccsc23)=O)C1 c1(C(=O)NCC2CCC(C(=O)OCC)C2)ccc(OC)c2cnccc12 c1(C(=O)NC(CNC(c2ccc(COC)s2)=O)C)cn2c(n1)CCC2 C1(NC(CCCC)=O)CCN(C(C2CCOC2C)=O)CC1 N(C1CN(C(=O)C=Cc2cccs2)Cc2ccccc21)C(C1C(C)C1C)=O N=c1[nH][nH]c2cc(C(=O)Nc3c[nH]nc3C(N3CCC34CCCCC4)=O)ccc12 Cn1nccc1C(C(=O)O)NCCC(=O)Nc1ccccc1 c1(C(N2CCC(CC)(CO)C2)=O)cc(F)c(C#N)cc1C C1(NC(c2c(C)cco2)=O)C2CN(C(=O)CC3CCCC3C)CC12 C(=O)(C(O)CC(N)=O)N(CCC(=O)NC1CC(CCC(=O)OCC)C1)CC=C N1(C(c2ccc(C(OC)OC)o2)=O)CCC(NC(=O)C(O)CC(N)=O)C(C)C1 Cc1nc(C)c(C(=O)NCC2(C(=O)NC3CCCC3C)CC2)s1 CC(C)CC(F)(F)C(=O)NC1CCC1NC(C1CCC(F)(F)CC1)=O C1(C(N(C(C)C)CCNC(=O)CCC(N)=O)=O)CCC2CC1CO2 C1(C(=O)NC(CC)Cn2cncn2)(CNC(=O)COCC(=O)OC)CCCCC1 N1(C(C2(C(=O)OCC)CC2)=O)CCC(CN(C(=O)C(C)n2cnnn2)C)C1 c1(NCC(CC)CCO)ncnc(NCC(C(C)CC)OC)c1C C1(NC(=O)C=CC2CCCCC2)CC2(C1)CC(NCc1cnc[nH]1)C2 c1(-c2cccc(C(C)=O)c2)cncc2sc(C(=O)Nc3ncc(F)cc3Cl)cc12 N1(C(C#CC(=O)N(C)C)=O)CC2CCCC(C1)N2CCOCCC(F)(F)F c1(C(C(=O)NCC(CO)NC(C2N(CCC)CCC2)=O)(C)C)ccc(C#N)cc1 N1(C(C2(OC)CCOC2)=O)CCC(C(=O)NCCCCCCF)CC1 c1(CC(N2C(CN(C(C3CNC(=O)N3)=O)CC)CCC2)=O)nccc(OC)n1 c1(-c2cn(C(COCC)C(=O)NC(C)(C)C(N)=O)nn2)cccc(O)c1 C(=O)(C#CC1CCOC1)NC1CN(C(C(C)CSc2ccccc2)=O)CC(F)C1 C(=O)(C(C)CS(C)(=O)=O)NC(CC)CNC(c1cc(C)c(C)nn1)=O C1(OC)C(NC(C2CC(N(C)C(C3OCCC3(C)C)=O)C2)=O)CC1(C)C C12(CC(N3CC(CCC)OCC3)=O)CCC1CN(C(C1(CO)CCCC1)=O)C2 N1(C(CC2C(C)=NNC2=O)=O)CCCN(C(=O)C(C(C)C)N2CCCCC2)CC1 C(=O)(C(O)CC(F)F)NC(CCCC)CNC(=O)C=Cc1cc(C)no1 Cc1cccc(C(=O)NCC(C)(C)CNC(c2cnc(O)c(Cl)c2)=O)c1Cl N1(C(C(c2n(C)ccc2)=O)=O)CCC(C=CC(N2CCCC(C)(C)C2)=O)CC1 C1(CN=C(NC(C2CC2C(F)(F)F)C)NCc2ccco2)CC2C=CC1CC2 N1(c2cccc(C(C)C)n2)CCS(=O)(=O)C(C)(C)C1 c1(CC(=O)NC2CC(NC(=O)CC34CCC(CC3)C4)C2)cc(O)nnc1O c1(OCCC)ccc(-c2cscc2C(=O)NC(c2ccc(C)cc2Br)=O)cc1F C(=O)(CC(O)C(=O)NC1CC1NC(C1(O)CC1)=O)OC(C)(C)C c1(C(N2CCN(C(CSCCC#N)=O)C3C2C3)=O)ccc2nc(O)oc2c1 c1(C(=O)NCC(C)(CO)NC(C2CCC(=O)N2)=O)cc(Cl)c(Br)[nH]1 CC(CC(=O)OC(N)=O)N(C(=O)CCNC(=O)C(C)CC1CCCC1)C C1(CC(N)=O)(NC(CCOCCC)=O)CCN(C(=O)C(CO)N(C)C)CC1 C(=O)(C(CC)(CC)CO)NCCC(C)NC(C=CC(CC)C)=O C1(C)(NC(C2CN(C)C2)=O)CN(C(=O)C=CCN(C)C)C1 CC(C)CC(O)C(=O)N1CCOC(CNC(C2CN(C)CC2C(F)(F)F)=O)C1 C(=O)(CS(=O)(=O)c1ccc(C(=O)NC2COCCC2c2ccccc2)cc1)NC c1(CC(=O)N(C2CCN(C(c3nnnn3C)C)C2)CC)cncn1C c1(NCc2n(C)cnn2)cnc(Cl)c(Cl)c1.N12CCN(CC1)C1(CC1)C2=O Cc1ccc(C(=O)NCC(C)(C)CCNC(=O)CC2CCC(C)C2)c(C)c1 c1(-c2cccc(C(=O)NCC)c2)cccc2c(C(=O)Nc3cncnc3)n[nH]c12 N1(c2ccc(CN(CC=C)CCO)cc2)C(=O)c2ccccc2C1=O c1(CNCC(O)Cc2ccccc2)ccc(OC(F)F)c(F)c1 C1(NC(CC(C)c2ccco2)=O)CC2CCC(C1)N2C(=O)C=CSc1nc[nH]n1 CC1(CNC(=O)Cn2ccccc2=O)CCCN(C(C2(Cl)CCCCC2)=O)C1 CCC(CC1CCCC1)C(=O)N1CC=CC1CNC(C1CS(=O)(=O)C1)=O C1(C(=O)NC2CC(C)(NC(C34CC(F)(C3)C4)=O)C2)CC2(CCOCC2)CO1 c1(CC)cc(C(N2CC(CN=c3[nH]nco3)C(CCO)C2)=O)ccc1C C1(CCCC)CN(C(=O)CC23CC(C2)C3)CCN1C(c1ncoc1-c1ccon1)=O N1(C(C2N(C(c3c(C)n(C)cn3)=O)C3C(O)CC2C3)=O)CC(=O)N2CCCC2C1 c1(C(C)C)c(CNC(=O)CN2CCOC(CC(C)(C)C)C2)ncnc1Cl Cc1cccc(C(=O)NCC2CC(CNC(=O)CCC3CC3)CO2)c1O c1(C(=O)NC2(CCOC)CCN(C(c3nc(Cl)c(Cl)s3)=O)C2)cc(C)nc(C)c1 C1(CCNC(C(c2cn(C)nc2)(F)F)=O)CCCCN1C(c1ccc(O)nn1)=O C1(CN(C(=O)CC=C(C)C)CC)CCN(C(c2c(C(F)(F)F)coc2C)=O)CC1 N1(C(C(C(COC)C)C)=O)CC2CCCC(C1)N2C(C1(Cl)CCCCC1)=O c1(C(C)C)n[nH]cc1C(=O)NCC1CCCC1NC(=O)CC(=O)Nc1nccs1 c1(C(=O)NC2CN(C(CCSCCC)=O)CC3C2C3)[nH]c2ccc(C)cc2c1Cl c1(CC(C)OC)nc(-c2ccc(C(C)(C)C)nc2)n(CC(N)=O)n1 CCC(CC)(CCNC(=O)C(c1ccccc1)=O)NC(=O)CCc1nccs1 c1(OC)cc(OC)c(NC(C2CC(F)CN2C(C2CC(=O)N2)=O)=O)cc1F C1(C(=O)NCCC(=C)CNC(=O)C=C2CCOCC2)CCCC(F)C1 C1(NC(c2ccc(Cl)cc2)=O)CCCC(C(=O)N(CCO)Cc2cccnc2)CC1 Cc1cnc(CNCC23CC2CN(C(c2cncn2C)=O)C3)nc1 C1(NC(C(C)(C)C(N)=O)=O)CN(C(c2cccc3nc[nH]c23)=O)C2(CCOC2)C1 CCCCC(CC)CC(=O)N1CC(NC(c2conc2C)=O)CC12CCCC2 N1(C(Cn2c(C)nnn2)=O)C(CNC(=O)C=CC2CCC2)CC2CCCCC12 Cc1c(C(N2CCCC2c2cnc[nH]2)=O)cn2[nH]cnc(=O)c12 c12ncccc1NCCS2.Cn1nnnc1SCCCCc1ccccc1 C=CCC(C1CC1)NC(=O)C(c1ccoc1)NC(C1CC1CCOC)=O C12(OC)CCCC1(C(N1CCC(C)C(N(C(=O)Cc3ccoc3)C)C1)=O)CCO2 C(=O)(C(C(F)(F)F)C(F)(F)F)NC1CCC(CCNC(=O)Cc2c[nH]nc2O)C1 N1(C(C2CCC(OC)C2)=O)CC2(CCN(C(c3cccc4nsnc34)=O)C2)C1 Cc1nn(C)c(F)c1C(=O)NCc1ccc(C(C)NC(=O)C(C)C(C)(C)C)cc1 C1(C(N(CC(CNC(CSC)=O)O)C)=O)CCn2c(C)nnc2C1 Cc1cc(C(=O)NCC2CC(F)CN2c2cc(C)nc(C3CC3)n2)nc(Cl)c1 c1(SC)ccc(CC(=O)NCCC(CNC(C2(O)CC(F)(F)C2)=O)OC)cc1 N1(C(C(C(C)C)O)=O)CCC2(CC1)CN(C(=O)C=Cc1ccco1)CCC2O c1(OCC)ccc2nc(N3CC4CC(NC(=O)CCCC(N)=O)C4C3)sc2c1 C(=O)(CCCCC(=O)NC12CC(NC(=O)CCCSC(C)(C)C)(C1)C2)NC c1(C(=O)NC2C(C)CN(C(c3ncc[nH]3)=O)CC2)ccc2nc(O)n(C)c2c1 C#Cc1ccc(C(=O)NC2CC3CC(NC(C4(O)CCSCC4)=O)C2C3)c(F)c1 CCCCCC=CC=CC(N1CCC1CNC(c1ocnc1CCC)=O)=O CC1(C)CCCC(C(=O)NC2C3CC(NC(c4cncc(N(C)C)c4)=O)CC23)C1 c1(OC)ccc(CC(N2CCN(C(c3occc3Cl)=O)CC2C)=O)c(F)c1 Cc1ncc(C(N2CC3CC(NC(C4CN(C(N)=O)C4)=O)C2C3)=O)cc1N n1(C(C(=O)OC)C)nnnc1C(c1cc(C(C)C)on1)NC1CC1C(F)(F)F Cc1cc(C(=O)NCC(C2CC2)N(C)C(C2CC3(CCC3O)C2)=O)cc(F)c1 C1(C(N2CC(N(C(c3ccc(NCCOC)cc3)=O)C)C2)=O)CCCC(C)(C)C1 C(CC(C)(C)CC(=O)N1CC(OC)C(NC(c2ccn(C3CCC3)n2)=O)C1)OC N1(C(C(C(C)C)CO)=O)CCC(F)(F)C(CNC(c2cnc[nH]2)=O)C1 C1(CC(=O)NC(CN(C(CSCC)=O)C)(CO)CO)CSc2ccccc2O1 C(CCCCC(=O)NC1CC(C)N(C(c2cc(N(C)C)ccn2)=O)C1)OC C1(C(=O)NC(CNC(C2CC2c2ccccc2)=O)C2CC2)CCCN1C(C)=O.CSC Cn1nnc2c1C(C(=O)NCC1(NC(=O)C3CC3)CCOC1)CCC2 C=CCCC(C(=O)NCC(CC)OC)NC(C1CCN1C)=O N1(C(=O)CC2CCCCN2C(C2C3CCCC23)=O)CCC(CO)C(O)C1 N1(C(CC=C(C)C)=O)CC2CCC1C(NC(=O)C1=C(C#N)CCC1)C2 C(=O)(C(C)(C)C1=CCN(C(=O)C(C)OC(CSCC)C)C1)N(CC)CC N(C1COCc2ccccc21)C(N(C(c1ccccc1)C)CCO)=O N1(C(C(C(C)(C)O)F)=O)CCC2(CCOCC2)C(NC(=O)CC2CCNC2=O)C1 c1(N(C)CC2(OC)CCOC2)nc(NCC(F)(F)Cl)c2ncsc2n1 c1(OC)cc(F)c2c(C(=O)NC(C)(CNC(C3(F)CC3C)=O)C(C)C)n[nH]c2c1 N1(C(C2(C)CCN2C(=O)Cc2cc(Cl)c(Cl)[nH]2)=O)CCC(C(N)=O)CC1 CN1N=C(CC(=O)N2CC(O)(CCNC(c3cn(C)nc3C(F)F)=O)C2)CC1=O N1(CC(=O)NC(C)CN(C)C(c2n[nH]cc2F)=O)CC2C=CC1C2 c1(OC)cccc(C(N2CCCCC2CN(C)C(c2ncc(Cl)s2)=O)=O)n1 c1(COC)cc(C(=O)NCC2(NC(=O)C(C3CCCCC3)F)CCOC2)cs1 c1(C(=O)NC2CC(C)CN(C(c3cnn(C4CC4)c3)=O)C2)ccc2n[nH]cc2n1 C(=O)(C(C)(C)C(C)(C)O)NCC1CC(O)(CNC(C2C(C)(C)CO2)=O)C1 C(=O)(C(O)C(CCC)NC(=O)C(C)(CC)OCC)N1CC(C#C)OCC1 C1(CC(=O)NC(C(=O)OCC)OC)(OC)CN(C(c2cnc(C(C)C)o2)=O)C1 c1(C(=O)NC2CCN(C(C=C(CCC)C)=O)CC2C)coc2cccc(Br)c12 C1(NC(C2C(OCC)CC2)=O)CC(C)(CNC(c2cnn[nH]2)=O)C1 N1(C(C2CC(SC)C2)=O)CCCC(C(N2CCCC3(C2)N=N3)=O)CC1 c1(C(N2CC(OCC)(CNC(c3[nH]c(O)nc3C)=O)C2)=O)cccn2nnnc12 c1(C(N2CCC(CCNC(c3c(C)[nH]cc3)=O)C2)=O)cnc(O)c([N+](=O)[O-])c1 C1(NC(C(C)(O)C2CCCCC2)=O)CCN(C(c2cn(CC3CC3)nn2)=O)CC1 c1(C(N(C(C(=O)OC)C)C)=O)ccn(CCNC(=O)C(C)n2ccnn2)c1 C12CCCC1C2.C1(C(=O)NC(c2ccc(-c3ccncc3)s2)=O)CC=CCC1 CCN=c1[nH]c(C(=O)NC2CCN(C(=O)Cc3csc(Cl)n3)CC2C)cs1 N1(C(C(C)(C)OC)=O)CCC(C)(CC(=O)NC2CCOC2(C)C)C1 C1(NC(c2c(C(N)=O)csc2)=O)CCN(C(c2coc(C3CCC3)n2)=O)CC1F C1(CNC(c2ccc3cnoc3c2)=O)Cc2ccccc2CN1C(=O)CO C#Cc1cccc(C(=O)NC(CO)C(C)NC(C2(CC(F)F)CCC2)=O)c1F C(=O)(CCCC(=O)NCC(C)CNC(c1oc(CC)nc1C)=O)NCC c1(C(N(CCNC(CC(C(C)C)OCC)=O)C(C)C)=O)cnn2c1CCCC2C N1(C(Cn2c(C)ccn2)=O)CCC(NC(C2CCN(C)S2(=O)=O)=O)CC(O)C1 C1(CNC(c2ccnc(S)c2)=O)CCN(C(=O)C(O)C2CCCC2)CC1O Cc1ccccc1C(=O)NC(c1cccc(C(C)O)n1)c1nnnn1C1COC1 N1(C(C2C(CC)C2)=O)CC(NC(c2cncc(C)n2)=O)CC2(CCC2)C1 c1(C(=O)NCC(C)(C(C)C)NC(c2nc(C)oc2)=O)cccc(F)c1C#N C(=O)(C(C(C)(C)C)C1CCCCC1)N1CCCC(CN(C(CCC(=C)Cl)=O)C)C1 Cn1cc(C(=O)NCC(=O)NC23CCCCC2C3)ccc1=O C1(NC(c2n(C)nc(CNC(=O)C(F)CC3CCC3)c2)=O)CCCC2(CC1)CC2 C1(C(=O)NCC(CC(=O)N(C2CCN(CC)CC2)C)C)CC(=O)OC1(C)C C(c1c(C)noc1C)=CC(=O)NC1CC(C(C)NC(C2(COC)C=CCC2)=O)C1 CC1(C)C(NC(=O)C=Cc2cc[nH]n2)CCN1C(=O)CCC(=O)Nc1nccs1 C1(NC(=O)Cc2cnn(C(F)F)c2)CCN(C(=O)C2=CCCSC2)CC1F N1(C(C(CC2CN(C(C3(C)CC=CC3)=O)C2)F)=O)CCCC(F)CC1 C(CC(C(=O)N(C(C)CC(=O)OC)C)NC(=O)C(C)N(C)C)SC c1(N(C)C)ccc(CNC(C2C3CC3CN2C(C2CC2(Cl)Cl)=O)=O)cn1 N1(C(c2cc(C)c(Cl)s2)=O)CC2CC1CN2C(C1CCCN1C(=O)C(C)(C)C)=O C1(C(=O)NC2(C(=O)O)CC(O)C2)CNc2ccccc2O1 Cc1cccc(C)c1OCCC(=O)NCC1(O)CC(NC(C23CCC2CC3)=O)C1 c1(C(=O)NC2C3CC(O)C2N(C(c2nn[nH]c2Cl)=O)C3)cccc2ccccc12 C(=O)(C(F)(F)C(C)(C)O)NC(C)CCCC(=O)NCc1cnn(CCO)c1 N1(CC)CC2CC1CN2c1cc(N(C)Cc2ncc(C)o2)nc(C(F)(F)F)n1 c1(C(N2CCC(CCF)CC2)=O)c[nH]cc(F)c1=O CC1(F)CCN(C(C2CC(O)CN2C(c2cccc(Cl)c2)=O)=O)C1 c1(COC)cc(C)c(C(=O)NCCN(CC(C)O)C(=O)CC2CN(C)CC2O)o1 CC(C)C(O)CC(=O)NCC1CCN1C(c1cnc(S)n1C1CC1)=O C=CC(C)(O)CC(=O)N1CCC(OCCNC(=O)C(C)(C)C2CCCO2)CC1 CC1CC(NC(c2nc(Cl)ccc2Cl)=O)CCN1C(C1CCS(=O)(=O)CC1)=O C1(C(N2CC(OC)C(NC(c3cc(C)nn3C)=O)C2)=O)Cc2cc(Cl)ccc2O1 N1(C(C#CC(C)C)=O)CCC2(CNC(=O)Cc3ccc(F)c(F)c3)CCCCC12 CCCS(=O)(=O)CC(=O)NC1CN(C(c2cnccc2Cl)=O)CC1C C1(n2ncc(C(=O)O)c2)CCN(C(=O)CN2CCCC(F)C2)CC1 c1(C(N2CCCC(OCC#C)C2)=O)ccc(F)c(Cl)c1F O=C(CC(F)(F)C(F)(F)F)NCC1(C2CC2)CCN(C(=O)CC23CCCC2C3)C1 c1(CC)ccc(C(=O)NCC(O)CN(C(=O)Cn2nc(C)oc2=O)C)nc1 N1(C(C(C)Oc2cccc(C)c2)=O)C2CCC1CC(CNC(C1(O)CCC1)=O)C2 CC(CCN=c1cc(Cl)nc(-c2cccnc2)[nH]1)NC(c1csc(Cl)c1Cl)=O C1(C)(C(=O)NC(c2ccccc2)C)CCCN1C(C1CCCSC1C)=O C(=O)(CCCS(C)(=O)=O)NC(C1CCN(C(C2(C(C)(C)O)CCC2)=O)C1)(C)C Cc1cccc2[nH]cc(CC(N3CCCC(NC(C4(O)CC4)=O)CCC3)=O)c12 c1(NC2CC(C)(C)OCC2)nccc(=NCc2cnccc2CO)[nH]1 C1(CC(=O)NCc2scc(C)c2)C2CCCC2N1C(c1ccc(C)nc1)=O N1(C(C2ON=C(C)C2)=O)CCC(O)(CN(C(=O)CCc2c(C)noc2Cl)C)C1 N1(C(C(COC)NC(C)=O)=O)CCC(=CCNC(c2coc(Br)c2)=O)CC1 c1(N2CC(C)(C3CC3)OCC2)nc(=N)[nH]c(=NCC(F)(F)C(C2CC2)C2CC2)[nH]1 C1(C(=O)NCCN(CC)CC)CCCN(C(C2(O)CCNCC2)=O)C1 C1(CNC(c2c(C)c[nH]n2)=O)CN(C(C2CCCCO2)=O)C(C)(C)C1 c1(OC)ccc(C2(C(=O)NCCCCCCN(C(=O)C(C)OC)C)CCC2)cc1 Cc1ccc(F)c(C(N2C3CCC(C3)C2C(=O)N(CCCO)C(C)C)=O)c1F C1(CCNC(CC2(N(C(C(CO)NC(=O)OC)=O)C)CC2)=O)CCC(C)CC1 c1(OC)cc(NC(C2COCCN2Cc2ccc(F)c(C#N)c2)=O)c(Br)cc1Br c1(C(N2CCC(N(C(=O)CC3CCC(=O)NC3)C)C2)=O)ccc(C#N)n1C C1(CC(=O)N(C(CNC(C2(C(=O)OC)CC2)=O)C2CC2)C)CSCCS1 c1(C(=O)NCc2c(CNC(C3C(COC)C3)=O)cccc2)ccc2n[nH]cc2c1 c1(N2CC(NC(c3cnc(C4CCN(OC(C)=O)C4)s3)=O)C2)ccc(N)cc1C C1(C(N(CC(CCC)C)C)=O)C=CCN(C(C2(OC(C)=O)CC2)=O)C1 c1(C(=O)NC2CN(C(C3C(OC)CCCC3)=O)C2)c(C)nc(C(C)(C)C)nc1O CC(C)C(O)CC(=O)NC1CCN(C(c2cn(C3COC3)nn2)=O)C12CC2 C1(F)(CNC(c2cccc(CCC)c2)=O)CCCN(C(C2C=C(C)CS2)=O)CC1 c1(N(C(C2CCN(C(CCCCC)=O)C2)=O)C)ccc(C)c(C)c1 c1(C(N2C3CN(C(Cc4c(C)noc4)=O)C(C3)C2)=O)ccc2nc[nH]c2c1 C(C)(C(=O)N1CC(CNC(C2(CCN(C)C)CC2)=O)C1)(C1CC1)OC C1(C(N2CCCC(NC(Cc3ncc(C)s3)=O)C2)=O)Cc2c(F)cccc2O1 c1(C(N2C(CC)C(C(N3CC4(CC4)C3)=O)CC2)=O)cnn2ccccc12 c1(C(N2CCC(NC(C(C)SCC)=O)CC2)=O)cc(F)c(Cl)cc1C C1(C(=O)NCCCN(CCCNC(C=CCN(CC#C)C)=O)C)CCCCO1 C1(NC=O)CCCN(CC(CN(C)Cn2nccn2)NC(=O)OC(C)(C)C)C1 CC1CC(C(N2C(CNC(C3(O)CCCC3)=O)CC3COCC23)=O)CC(C)(C)C1 N#Cc1c[nH]c(C(=O)NCc2ccccc2CNC(C2CC2[N+](=O)[O-])=O)c1 C1(NC(C=Cc2ncn(C)c2)=O)CC2CC1N(C(C1(C)CC1(F)F)=O)C2 c1(C(=O)NC2CN(C(C#CC(=O)O)=O)CC(F)C2)n[nH]c2cccnc12 CCC(CC)C(=O)N(C1CCC(NC(=O)CC(c2cccs2)NC(N)=O)CC1)C c1(OC)nscc1NC(C1OCCC1CNC(C1(NC(N)=O)CC1)=O)=O C(C(C)(C)C(=O)NCC1(F)CCN(C(C2CC(=O)N(C)C2)=O)C1)OCC C1(C(=O)NC(C2CCOCC2)C)(CC)CCN(C(=O)C(C)SC(C)C)C1 C(=O)(CC(C)C(=O)N1CCOCC1CCNC(c1c(OC)cccc1Cl)=O)OC c1(C(C(=O)NC)N(C2CC2)Cc2cccc(C(C)C)c2F)cc2ccccc2o1 C1(CNC(c2c(C)nc(O)s2)=O)CC12CCN(C(C1CC(C)(F)C1)=O)CC2 CC1(C)CC(NC(c2ccc(F)c(I)c2)c2nnnn2CC2CC2)C12CCC2 c1(COCC)nc(N2CCC(C)(NC(=O)Cc3ccon3)C2)cc(C)n1 N1(C(Cc2c(C)cco2)=O)CC(C)CN(C(c2n[nH]c(=N)[nH]2)=O)C(C)C1 N1(C(C=COCC)=O)CCC(CCNC(c2ccc(S(C)=O)cc2)=O)C(F)(F)C1 N1(C(C(CC=CC)NC(=O)CNC(=O)OCC)=O)CCOCC(CO)C1 c1(C(=O)Nc2nc(C3CCCNC3)cs2)ccc2c(c1)CC2 C(C(COC)CC(=O)NC1COCC1C(N1CCC1CN=[N+]=[N-])=O)OC N1(C(=O)CCn2cncn2)CC2CCN(Cc3cc(Cl)c(Cl)c(Cl)c3)CC2C1 C1(CC(=O)NCCC2CN(C(C3CCC(=O)NC3)=O)C2)CC2(CCC2)CCO1 N1(C(C(CC)c2ccccc2)=O)CCC(C2(NC(c3ccc(CO)nc3)=O)CC2)C1 Cc1nc(NC(C)Cc2ncccc2C)cc(NC2CCCCCC2)n1 c1(CNC(C(=O)NC(c2ccnn2C)CC)=O)cccc2c1OCCCO2 C(N=c1[nH]c(N2CC3CC2C3)nc2c1CCCCCC2)c1cn(C)[nH]c1=N c1(C(N2CC3(CNC(C45CSCC4C5)=O)CC2CO3)=O)ccc(F)cc1F C(=O)(CC(c1ccccc1)NC(=O)C(F)(F)F)NC(CC)CNC(=O)C(C)OC N1(C(CCCC=C)=O)CCC(CNC(=O)C(CCC)N(C)C)CC1C c1(COC)ccccc1C(=O)N(C)CC1CCCN1C(=O)CCc1cnn(C)c1 CCCCCC(O)CC(=O)NC1CC2CN(C(C34CC3C4)=O)CC2C1 C1(CN(c2cc(NCC34CCCC3CCC4)ncn2)C)CCc2c[nH]nc2C1 N1(C(C(C=C)OC)=O)CCC(C2CC2)C1C(=O)NC(COCC)C(C)C CC1(CS(=O)(=O)OCC2CC(F)(F)C2)COCCN1 n1(CC)ccnc1C=CC(=O)NC(C1CCCC1)CNC(c1ncoc1C)=O c1(C(=O)NC(C2CCC(F)(F)CC2)CC)cn2c(n1)CCC2 C1CCC(CO)NC(=O)C=C(C)CC(=O)N1.C(=O)(C(C)(F)F)N=C(C)C CC1(CNC(C2CCOC2CNC(C2(CCN(C)C)CC2)=O)=O)NC(=O)NC1=O CC1(CNC(=O)C(=O)NCC2CC2)COCCN(C(=O)C=Cc2ccc(Cl)s2)C1 N1(C(C(C)NC(C)=O)=O)CCC(O)C(C(N2CC(O)CC2CO)=O)C1 N1(C(C(COCC)(C)C)=O)CCN(C(=O)CCC=CBr)C(CF)C1 Cn1cnnc1C1CCN(CC(O)Cn2cccn2)C1 c1(C(=O)NC2CN(C(C(C)NS(CCCC)(=O)=O)=O)C2)cc(Cl)ccc1C c1(NC(CC)C(C)C)ccc(S(=O)(=O)N(CCC(=O)NC)CC2CC2)cc1Cl C=CCCC(CC(C)C)C(=O)N1CC2CC(N(C(=O)CNC(N)=O)C)C1C2 CCC(C)C(CC(=O)N(C)CC1CCCN(C)C1)NC(=O)C(C)(C)n1cccn1 C(CC(C)CC(C)(C)C)NC(CN(C(c1c(C(C)C)nco1)=O)C(C)C)=O c1(C(=O)NC(C2(CNC(c3ccc[nH]3)=O)CC2)C)ccc(F)c(Cl)c1F N1(C(CN(C)CC)=O)CCCC2(CCN(C(=O)Cn3nc(C(F)F)cc3C)C2)C1 c1(N(CCC(N2CC(O)(COC)C2)=O)CC)ccccc1[N+](=O)[O-] c1(SCC)ccccc1C(=O)NCC1CC1NC(=O)CNS(=O)(=O)NC.C(N)=O N12CCCCC(C1)C2=O.C1(CC(=O)Nc2cncc(CC)c2)CCCS(=O)(=O)C1 C1(NC(=O)NCC(=O)N(C)C)CCN(C(C2CC2(C)C)=O)CC1c1cccnc1 Cc1c(NCCCCC(C)C)ncnc1N(C)CC1CCC1 C1(C(N2CCC(CCNC(c3ncncc3Cl)=O)C2)=O)CCC2(CCOCC2)C1 c1(CCC)nc(C)c(C(=O)N(CC(C)(C)NC(=O)CN(C)C(C)=O)C)s1 C=CC1CN(C(C2CNC(=O)CN2C(C2CCC3(CCC3)C2)=O)=O)CC1O C=CCC(C(=O)N(C1(C(N2CCN(C)C3CC23)=O)CCC1)C1CC1)C(C)C c1(CC(C)C(N2CCC(NC(=O)C(C)(C)C)C(O)C2)=O)ccc(O)c(O)c1 N1(C(C(C)(C)C2CCCO2)=O)CCC2(CCCN2C(C2CC3(CCC3)C2)=O)C1 N1(C(C=CC(=O)OCCCC)=O)CCC(F)C(NC(=O)Cc2csc(Cl)n2)C1 n1(CC)nc(C(=O)NC2(C)CC(NC(=O)Cc3ccnn3C)C2)c2c1CCOC2 c1(N2C(=O)C3CC(=O)N(C3)CC2)ccc(N)cc1Cl.C12(F)CN(C1)C2=O.CNC N1(C(C(C)OCCN(C)C)=O)CC(F)(F)CC1CNC(C1CCCCN1N=O)=O c1(OC)ccc2[nH]c(=NCc3csc(C4CC4)n3)[nH]c(=NC3COCC3C)c2c1 N1(C(CCC(C)C)=O)CCCC2(CCCN2C(=O)CC2CCC(C)(C)CC2)C1 c1(C(=O)NC(c2ccc(F)cc2)C(F)(F)F)csc(C2=COCCC2)n1 Cc1cccc2c1CN(C(C1(C3CC3)CN(C(=O)C(C)CC(C)(C)C)C1)=O)C2 c1(OC)ccc2nc(NCCNC(C3CN(C)CCN(C)C3)=O)c(C#N)cc2c1 N1(c2nccc(OCC)n2)CC(NC(=O)C=CBr)CC12CCOCC2 c1(C(=O)NCC2N(C(C(C)OCC)=O)CCCC2C)cc2cccc(F)c2o1 C1(CNC(=O)NC2CCN(C(C34COC(CF)(C3)C4)=O)CC2)CCCC1C1CC1 c1(CCC(=O)N(CCCNC(c2c(CCC)n[nH]c2)=O)CC)ccc(OC)nc1 N1(C(CC2C(C)(C)OCC2)=O)CCC(F)(C(=O)NCCN2CCC(O)CC2)CC1 c1(C(N2C(C)CN(c3nccc(Br)n3)CC2)=O)cc(F)c(F)cc1[N+](=O)[O-] C1(OC)CCCCC1C(N1CCC(N(C(=O)CCC2CCCC2)CCO)CC1)=O N1(CCC(=O)NCC(C2CCCC2)NC(=O)CC2CCC2)CCNC(=O)C1 N1(C(C2(C)CCCN(C(CCN(CCC)C)=O)C2)=O)CCCC2(C=CCO2)C1 c1(C(=O)NCC23CCC2CN(C(c2ccc(Cl)cn2)=O)C3)nccn2nccc12 C(=O)(C(C)S(=O)(=O)C(C)C)N1CC(C(C)C)N(C(=O)C#CC2CCC2)CCC1 Cc1cccc(C)c1OC(F)F.c12ncnc(c1C)CN2CC(=O)NCC(F)F N1(CC)CC(NC(=O)CC(C)(C)NC(C2OCCC2C(C)C)=O)C(C)C1 C(=O)(C(CNC(=O)C(=O)NC)C(C)(C)C)NC1C(CC)C1 c1(CC(=O)NCCCCCNC(C2(C)CC(=C)C2)=O)cccc(C(C)C)c1 CONC(=O)C(=O)N(C1CCCN(C(=O)CCN2CCCCC2)C1)CC1CC1 C(CCCCC(=O)NC(C)(CNC(c1ncn2c1CCC2)=O)CO)OCC N1(C(Cc2cccc(OCC)n2)=O)CC(NC(=O)C(F)CC2CC2)CCC(O)C1 N1(C(C2C=C(C)CS2)=O)CCC(C(CO)NC(=O)C(C)Cc2cnc[nH]2)CC1 N#Cc1cc(NC(=O)CC2CN(C(c3cc(O)c(O)c(Cl)c3)=O)C2)ccc1Br C(=O)(C(C)(O)CCN(C)C)N1C2(CNC(C3CCN(CC)C3)=O)CC(C1)C2 c1(CN2CC(O)(CNC(c3ccc(F)c(Br)c3)=O)C2)cc(F)c(O)cc1F C1(COC)(NC(=O)CCC(C)(C)C)CCCN(C(C2CC2c2ccccc2)=O)C1 C(=O)(CCC(C)(C)N(C)C)NCC(C)(CNC(=O)C(C)C(C)(C)C)OC C1(OC(C(=O)NCC2CN(C(CNC(C)=O)=O)C2)C)CCCCC1 C1(NC(c2[nH]cc(C(C)=O)c2)=O)CS(=O)(=O)CC1NC(c1coc(C(F)F)c1)=O c1(C(C)(C)C)cccc(CC(N2CCC(C(F)(F)F)(C=CC)C2)=O)c1 C1(C(N2C(CN(C)C(c3ccc(C(F)F)o3)=O)COCC2)=O)CCCC(F)(F)C1 N1(C(COCC)=O)CCCC(C)(C)C1C(=O)Nc1ccc(N(C)C)nc1 c1(C(=O)NC(C2CN(C(=O)C(=O)Nc3ncc[nH]3)C2)C)ccc(S(C)=O)cc1 C(CC1=CCN(C(=O)CNC(C2CC2C)=O)CC1)NC(c1c(C)ncn1O)=O N1(CCC(=O)NC(C)CC(C)NC(=O)CN2CCCC2=O)CCCS1(=O)=O c1(C(=O)NOCC2CC2)cccc(CNC(c2cc(-c3ccc(F)cc3)[nH]n2)=O)c1 CCCC(CN=c1[nH]c(N2CCC(Br)=C(C)C2)nc2c1SCC2)OCC C#Cc1nc(C(=O)N(C(CNC(C2CSCCS2)=O)C2CC2)C)cs1 C1(C)(C(=O)OC)CCN(C(c2cccc(I)c2)C(=O)NCc2ccccc2)C1 Cc1c(CC(=O)NCc2cc(C(=O)NCC3CCCC(O)C3)cs2)ncn1C N1(C(CC(CC)(C)C)=O)CC(CO)C2(CCN(C(=O)C(C)C(C)COC)CC2)C1 C1(CNC(C(C)Cn2cccn2)=O)CCCCCN1C(C1CC2(CSC2)C1)=O N1(C(CCCCNC(C)=O)=O)CCC2(NC(C3CCC(C)C3)=O)CCCC12 N1(C(C(C)=C2CCC2)=O)CCCCC(N(C)C(c2ccc(F)s2)=O)C1 Cc1cc(C(N2CCC(F)C(NC(c3cn(C)nn3)=O)C2)=O)nc(O)n1 C1(C(=O)NCC(C)(O)CNC(=O)CSc2ccc(F)cc2)CCCCC(F)(F)C1 c1(C(=O)NC(C)CNC(c2cccc(=S)n2O)=O)cc2n(n1)CC(F)C2 N1(C(C2CC(S(C)(=O)=O)C2)=O)CCC2CCCC12CO C(=O)(CCCC(=O)N1CCC(NC(c2csc(C3CCCCC3)n2)=O)C1)OC N1(C(c2c(C)cc(Cl)cc2)=O)CC2C(C1C(N1CC(O)C1)=O)C2(C)C Cc1coc(C=CC(N2CC3CC3(NC(=O)CCCCN(C)C)C2)=O)n1 c1(C(N2CCCC(C)(NC(=O)CCP(C)(C)=O)C2)=O)cccc2ccsc12 CCCC(CNC(c1ccsc1)=O)C(=O)N(C1CCOCC1)CCC C1(NC(COCCC#C)=O)CC(O)CN(C(c2ccc(O)c(CC)c2)=O)C1 CC1CC(=O)NCC1C(=O)NC1CN(C(=O)CN2OC(C)(C)CC2=O)C1 C1(CCNC(c2c(C)onc2)=O)CC(F)(F)CN1C(=O)COCc1cccnc1 C#CCC(CC#C)C(=O)NCC1(C(N)=O)CN(C(=O)C(COC)N(C)C)C1 CC(O)(CNC(=O)C(C1(O)CCCC1)F)CNC(C1(C(F)(F)F)CCC1)=O c1(C(=O)NC2C3CN(C(CCOCC)=O)C(C3)CC2)csc2c(C)cccc12 C1(O)(CN(C(=O)CC2CCCSC2)C)CCN(C(=O)COC2CC2(F)F)CC1 c1(N2CCC(C(CC)C)CC2)nc2c(c(=NCCC3CCCCO3)[nH]1)CCC2 c1(C(=O)NC(C2CCOC2)CNC(C(=CC2CCCC2)C)=O)ccnc(C)c1C CCC(F)(F)C(C)(C)C(=O)NCC1C=CC(NC(c2ccc(=N)[nH]c2)=O)C1 CN1CC2(CC2)CC1C(N1CC(O)(C(C)(C)CNC(c2cn[nH]c2)=O)C1)=O N1(C(c2cc(C)c(C)s2)=O)CCC2(CC1)CN(C(=O)C=CS(C)=O)C2C(C)C C(=O)(Nn1cnnc1C)C1(F)CCN(C(C(C(C)(C)C)OC)=O)C1 N(C1C(=O)Nc2c(C)cccc21)C(C1CCN(C(c2scc(C)c2)=O)CC1)=O C12(C(=O)NCCCN3CCCC3)COCC1CN(CC13CCCN(CC1)C3)C2 c1(C(=O)NC2(C(=O)Nc3cc(CC)c(C)cc3)CC2C)cccc2nccn12 N1(C(C(C)=C(C)C)=O)CC(NC(=O)Cc2cnn(C(F)F)c2)CCC1C C1(CNC(c2c(C)cnnc2O)=O)CCCC2(CN(C(c3ccsc3C)=O)C2)O1 c1(NC(=O)NC(c2cccc(Cl)c2Cl)CO)cnccc1[N+](=O)[O-] N1(C(C(c2scc(C)n2)C)=O)CCOC(C(C)NC(c2nccn2C)=O)C1 O=C(CCC(=O)N1CCOCC1)NCCc1cn(CC)nn1.C1(CC=CC)CCC1 C1(C(=O)NCC2C(C)(C)CCO2)CC2CN(C(=O)CC3CCC(=O)CC3)CC2C1 CON(C(=O)C1CCCN(C(=O)CCn2ccnc2C)CC1)C1CCC1 N1(C(CC(C)F)=O)CCOC(CN(C(=O)C(N2CCOCC2=O)C)C)C1 C(c1c(C)coc1C)=CC(N1CCC(C(CNC(C(CC)=CC)=O)C)CC1)=O C1(CC)CCN(C(=O)C(C)C2CCCC2)C(C(=O)Nc2cncnc2O)C1 C1(CCC)CCCCN1C(C1C2CCCCC12)C(=O)NC1CC(F)(F)C1 c1(C(=O)NC(CC)CNC(C2CC=CC2)=O)csc(=NC2CCCCC2)[nH]1 C1(C(C)C)CN(C(C2CCOC2CNC(c2ccc(O)nn2)=O)=O)CCCO1 c1(C(=O)NC2CC(CNC(C(C)(C)CF)=O)C(O)C2)cc2c(cc1Cl)NCC2 CCCCCCC(C)C(=O)NCc1ccc(CNC(c2ncoc2CC)=O)cc1 N1(C(C(C)OCCOC)=O)CC2CC2(CNC(=O)CNC(=O)CCCCO)C1 N1(C(CC(C(=O)OC)C)=O)CC2(C1)SCCC2NC(=O)Cc1ccn(C(F)F)n1 C#CCC(C(=O)NC(C=C)C(F)(F)F)NC(c1cnn(CC)c1)=O CC(CC(=O)NC1CCN(C(=O)C(C)(C)S(C)(=O)=O)C1)C(C)(C)C C1(NC(C2(C)ON=C(C)C2)=O)CN(CC(O)COCC2CCCC2)CCC1C N1(C(COC)=O)CCC2(C1)CN(C(=O)CN(C)S(=O)(=O)N(C)C)CCO2 c1(C(=O)NC2C(SC)CN(C(C3(C)COC3)=O)C2)cccc2cnccc12 N1(C(=O)OCC)CCCC(c2nc(C(=O)OC3CC3CC)cs2)C1 N1(C(c2c(CC)ncs2)=O)CCCCC(CNC(=O)Cn2nnnc2C2CC2)C1 N1(C(C2CCc3n(cc(C)n3)C2)=O)CCc2cc(Br)cc(F)c21 CCC(C)CCC(O)CC(=O)NCC1CCCCN(C(=O)C(C)(C)C(C)C)C1 c1(CN2C(C(=O)NC3C(NC(c4csc(O)n4)=O)COC3)CC2)cccc(Cl)c1 C1(NC(Cc2c(C)cccn2)=O)CCCCN(C(=O)C(C)OC2CCCCC2)C1 c1(C(=O)Nc2c(C)nc(-c3cccc(CN(C)C)c3)cc2)ccc2ccoc2c1 c1(C(N2C(CNC(C(C)SCC)=O)C3CCC2C3)=O)cncc2ccsc12 C1(CC)C(C(=O)NC2CC2c2cncs2)CCCN1C(c1scc(C)c1C)=O C(C(C)(C)C)=CC(=O)NCC1(CN(C)C(C2CC(N3CC(O)C3)C2)=O)CC1 O=C1NCCN(Cc2cc(F)cc(F)c2)C1c1ccccc1F C1(C2(O)CCOCC2)(C(=O)NC2C(NC(c3cc(C(C)C)on3)=O)COC2)CC1 C(CC(C)(C)CN)N(C(C(C)n1cccn1)=O)CCO Cc1cc(C(N2CC3CN(C(c4cc(=O)cc[nH]4)=O)CC3C2)=O)cc2c1CCC2 N1(C(c2c(C)oc(C)c2Br)=O)CCC2CCN(C(=O)CCCN(C)C)C2C1 c1(C(=O)NCCCCC(C)NC(COCC=C)=O)ncn2c1CCCC2 N1(C(C2(C#N)CCCCC2)=O)CCCCCCC1C(=O)NCCCCCCO CC(C)CS(=O)(=O)CCC(=O)N1CCCC1C1CCCN1C(c1cccnn1)=O N1(C(CCCNC(=O)OC)=O)CC2OCCN(C(=O)C(C)CC3CCCCC3)C2C1 N1(C(CCc2n(C)ccn2)=O)CC2CC1CCC2NC(=O)COCC1CC1 CC(CCC(C)(C)C)C(=O)NCC1CC1CC(=O)NC1CN(C)C1 c1(CN(C(c2n[nH]c(C)c2Cl)=O)C)ncc2c(n1)CCOC2.C12CCCCN1C2 C1(CNC(CCCC#C)=O)CC2(CCC2)CN1C(=O)Cc1cc[nH]c(=N)c1 c1(CCC(=O)NC2CCC(NC(C(=O)N(C)C)=O)C2)ccc(NS(C)(=O)=O)cc1 C(CC(CC)C(=O)N1CC(O)(CCNC(=O)C(C(C)C)NS(N)(=O)=O)C1)=CC c1(CNC(CC2C(C)(C)C2)=O)cccc(CNC(C2CC23CCC3)=O)c1 Cn1ncc2c(C(=O)NC3C4CCC3N(C(C3CC35CCCC5)=O)C4)ccnc12 C1(CNC(C(C)N(C)C)=O)CN(C(=O)C(C)n2cccc2)CCC1C c1(C(=O)NCc2cncc(OC3CC3)c2)cc2cccn2c(O)n1 CC1=CCC(C(=O)NC2C=CCN(C(=O)C(C)(C)n3cccn3)C2)CC1 Cc1c(C(=O)NCC2CCN2C(=O)C(C)CC2CC2)cncc1Br C1(C(=O)NC(C)C(=O)NC2CCCC2)C=CC(C(=O)NCC(C)SC2CCC2)C1 CC1CCN(C(c2cnc(O)n(C3CC3)c2=O)=O)C(C)C1NC(c1cc[nH]c1)=O C=CCC(F)(F)CN(C(C1CCCCC1)C(=O)NCCC1(C)CC1)C Cc1cnc(C(=O)NC2CCC(CNC(=O)C(C)(C)c3ccnn3C)C2)nc1 C1(C(N(C)CC2N(C(C3C(C)C3)=O)CCOC2)=O)CCc2nnnn2CC1 C1(C(N2CC3COCC3(C(N3CC(F)C3)=O)C2)=O)CCc2ccccc2C1 c1(C(C(=O)NC(C)C(C)NC(c2cnc(C(N)=O)s2)=O)=O)cc(F)cc(Cl)c1 c1(C(N2CCC(C)(NC(C(C)CC3CC3)=O)C2)=O)cc(S(N)(=O)=O)c[nH]1 C1(NC(C=COCC)=O)CCN(C(=O)CC2CC(CC)=NO2)C1C C#CC1CC2CCC1N(C(C1C3CCN(C(=O)C=Cc4ccncn4)CC13)=O)C2 C12(C(=O)NCCC(C)NC(=O)CCCC3CCCCC3)CC3CC(C(=O)N1)C2C3 C1(OC)CC(CO)N(C(=O)C#CCNC(=O)CC(C)N(C)C)C1 C12(NC(N3CCCC(Cc4nnc5ccccn45)C3)=O)CCCC1CC(F)(F)CC2 CCCCC(C(=O)N1CCCC(C)C1CNC(C1CC(C)C12CCC2)=O)N(C)C c1(CC(=O)NC(CNC(C(C2CCCC2)OC)=O)(C)C2CC2)cccc(F)c1 Cn1ccn2ncc(C(=O)NC3CCN(C(=O)CNC=O)C(c4ccccc4)C3)c12 CN1CCN(C(=O)C(CNC(c2ccnnc2O)=O)N(C)C)C(CCO)C1 N1(C(c2c(C)nncc2)=O)CC2CCC(N=c3[nH]c4cc(Cl)cc(Cl)c4o3)C2C1 c1(C(N2CC(CNC(=O)C(O)C3CC3)C(C(F)(F)F)CC2)=O)nccn2ccnc12 N1(C(=O)C(F)(F)C2CCNC2)CC(O)CC1c1cccc(F)c1 c1(CC)ccc(C(=O)NCCC2(CNC(C3CCOCC3C)=O)CC2)cc1 c1(C(=O)NCC(CNC(=O)Cc2cccnc2)OC)c(Cl)cccc1Br C1(CNC(C(C)=C(C)C)=O)CC2CCC1N2C(=O)C1=C(C)OCC1 N1(C(C(C)(C)SC)=O)C2CCC1C(C)C(NC(c1cc(C)oc1C)=O)C2 C(=O)(CC(F)(F)C(F)F)NC1CN(C(c2ccc(N3CCN(C)CC3)cc2)=O)C(C)(C)C1 C(CCNC(c1cccc(Cl)n1)=O)(C(C)C)NC(C1(C(=O)OC)CC1C)=O C1(CCNC(C2CC(SC)C2)=O)CC(F)(F)CN1C(C1CC2(C1)CC(C)C2)=O c1(CNC(NCC2CCCC(F)C2)=NCCF)cc2ccccc2[nH]1 CC(CCCCNC(C1CCCCN1C1CCCC1)=O)NC(C1CNC(=O)N1)=O c1(OC)cncc(C(=O)N(C(CNC(=O)C(F)C(C)(C)O)C2CC2)C)c1C c1(OCC=C)ccc(CC(N2CCC(NC(C3CCCO3)=O)C2C(C)C)=O)cc1 c1(N2CCC(OC(C)(C)C)CC2)nc2c(c(=NCC3C(C)(C)C3(F)F)[nH]1)COC2 c1(C(=O)NCC(O)CNC(c2coc(CC3CC3)n2)=O)csc([N+](=O)[O-])c1 C1(C(N2CCC(O)(CN(C)C(C3SCCCS3)=O)CC2)=O)CNC(=O)C(C)(C)C1 C(=O)(CCC1CCc2ccccc21)N1CCCCC(NC(C2CC(=O)N2)=O)C1 C1(NC(c2nc(C)nn2C)=O)CN(C(=O)C=C2CC2)CCC1C C1(NC(c2n(CC)ccn2)=O)(COC)CCCN(C(C2CCCN2C=O)=O)C1 c1(C(=O)NC2CC(C)N(C(c3ccc(C(F)F)cn3)=O)C2)cc2ccsc2s1 C(CC(C)C(=O)NC1CCC1C(N1CC(OCCF)C1)=O)=CC C1(CC)CN(C(c2ccccc2C)C(=O)NC)C(C)CO1 C1(NC(C2OCCO2)=O)CCN(C(=O)COc2ccc(F)cc2)CC1F c1(C(N2CCN(C(C3N(CC)CC3)=O)CC2)=O)ncsc1S(N)(=O)=O c1(C(=O)NC(CC(=O)NCCC(C)N2CCCC2)C(F)F)cc[nH]c2nccc1-2 C1(NC(c2cnc(CCCC)s2)=O)C2CCN(C(=O)CC(C)C)C2C1(C)C N1(C(c2ccnc(-n3cncn3)c2)=O)CCCN(C(C2CC2CF)=O)CC1 O=S1(=O)c2ccc(cc2Cl)N1.C1(COCCNCCCO)CCCO1.c1(SC)ccsc1 C1(CN(C(CC2(C=C)CCC2)=O)C)CN(C(C2CSCCS2)=O)CCO1 C#CC1COCCN1C(=O)C(C)(C)C1CCN(C(=O)CCCC2CC2C)C1 CC(C)S(=O)(=O)c1ccc(C(=O)NCCC(C)NC(C2CC(C3CC3)C2)=O)cc1 n1(C(CC)CC)nc(-c2ccc(SC(C)(C)C)nc2)nc1C(C)(C)CC N1(NC(=O)NC2C(C)COC2)CCN(Cc2ccccc2)CC(C)(C)C1 C12(NC(=O)C3CC3)CCN(CC1)C2=O.C1(CC)CCC2CC12 c1(C(CC)NC(=O)C(CCC)NC(N)=O)ccc(OCC)c(Cl)c1 C(=O)(C(CC(C)C)ONC(c1ccccc1C#N)=O)N1CCC(CC(=O)OC)C1 Cn1cc2c(n1)CC(C(N1CCC(F)(CNC(c3ccnc(O)c3)=O)C1)=O)CC2 c1(CC)ccc2c(c1)C(CC(=O)N(CCCN(C)C(c1ccsn1)=O)C)C(=O)N2 c1(CC)cnc(O)c(C(N2CC(CNC(=O)CCCCc3ccccc3)C2)=O)c1 c1(C(=O)NCC(CC=C)NC(c2nnn(CC(=O)OC)c2N)=O)cc2occc2n1C c1(NC(CC2CCCN(C(CCc3c(C)cccn3)=O)C2)=O)ccc(F)cc1Cl C(N=c1[nH]c(N2CCC(NC3CCC3)CC2)nc2ccsc12)C1CCN(C)CC1 c1(C(=O)OC)cnc(C(=O)NC2(CNC(c3cnc(C)s3)=O)CCCC2)c(N)c1 c1(C(C)C)nsc(NC(=O)C(=O)NC2(n3cc(Br)nn3)CC2)n1 c1(C(=O)NCCC2CCCN(C(CC(=C=C)C)=O)C2)cc(OC)cc2c1OCC2 C(CCC(=O)N1CCC(Cn2cc(C3(C)CCCO3)nn2)C1)CC(CC)N C(c1cccc(CO)c1)=CC(N1C(CO)CCC1c1ccccc1)=O C1(NCC(C)C(=O)O)CC2(COC(C)(C)C2)C1 N1(C(Cn2ccc(C)n2)=O)CCOCC1CNC(=O)CCc1ncccc1C N1(CC)CCC(C(=O)NC23CC(NC(=O)C(c4ccccc4)F)(C2)C3)CC1 n1(CC(=O)NC2C(NC(CC3CC(OCC)C3)=O)CCC2)cc([N+](=O)[O-])cn1 C1(N(C)C)(C(=O)NCC(c2cccnc2)NC(C2(C)CC(F)C2)=O)CCOCC1 N1(C(C23CCC(OC)C2C3)=O)CCC(NC(C2CCCCN2C(C)=O)=O)C12CC2 N(C(=NCCCCl)N1CCC(C)(OC)C1)CCc1c(OCCOC)cc(C)cc1 c1(CN(C(=O)C(N2CCc3cccc(Br)c32)=O)CCC)cc(Cl)cc2c1OCC2 CCC(C)(CNC(c1cscc1Cl)=O)NC(=O)C(C)OCCOC C1(OC)CN(C(=O)CSc2nnc(C)s2)CC1NC(C1CCOC1C(F)(F)F)=O C(=O)(C(C)C(=O)NC1CCCC1NC(C1(c2cccc(Br)c2)CC1)=O)OC Cc1ccnn1CC(=O)NC(C)CCCNC(c1cc(C2CC2)no1)=O n1(CC)nc(C2CC2)cc1C(C(=O)NC(C)C(=O)OC)N1CCCC1 c1(C(=O)NCCC2(OC)CN(C(c3ccccc3C)=O)C2)c(C)ncn(C)c1=O Nc1ccc(Cl)c(C(=O)NCC2CCCN2C(c2cc(CCO)on2)=O)c1 CC1=NOC(CC(=O)NCC2CC(CC(=O)NCC3(CO)CCC3)C2)C1 C1(NC(C2CC3CC(=O)C2C3)=O)CC(C(=O)N2CC3(CCCO3)C2)=CC1O c1(CC(=O)NC2(C)CC(NC(C3CCCCCCC3)=O)C2)ccc2c(c1)COC2 C(C#CC(=O)NC(C)C(C)(C)OC)NC(COC(C)=O)=O c1(C(N2CC(C)(CCC(=O)NCC(O)C3CCC3)C2)=O)sccc1C#N C(C)(CCC(=O)NCC1CCCCC1C(=O)NCCS(C)(=N)=O)OCC C1(CC(=O)NCCCOCCNC(CNC(=O)OC)=O)CCC2CC12 N1(c2cc(C#N)ncn2)CC2(CCC(NC(=O)CN3CCCC3)C2)C1 Cc1ccc([N+](=O)[O-])cc1NCc1ccncc1CN1C(=O)CCc2ccccc21 c1(C(N(C)CC2(O)CCCN(C(CC(C)SC)=O)C2)=O)n[nH]c2ccc(F)cc12 C=CC(CC)CC(=O)N1CC(CNC(c2cnc(COC(C)(C)C)s2)=O)C(C)C1 N1(C(C(C)CSCc2cccnc2)=O)CCN(C(=O)C(F)(F)CC2CC2)CC1 CCCC(C(=O)NCC1CCC(C(N2CCC(F)(CO)C2)=O)O1)OC n1(CC)ccc(C(=O)NCC(C2CC2)NC(=O)CN2CCCC2C)cc1=O CCCC(CC(C)C)C(=O)N1CC(O)CC1CC(=O)NC1CCC([N+](=O)[O-])CC1 CC1C(NC(=O)CCOCCNC(=O)C=C2CCC2)CCN1C N1(C(CC2CCCC(C#N)C2)=O)CC2CC1CN(C(c1coc3c1CSC3)=O)C2 C1(C(=O)NCCC(F)Cn2cc(CCN3CCOCC3)nn2)CCCCC1OC c1(CC)ccc(C(=O)NCC2CCN(C(=O)C=C(Cl)Cl)C2(C)C)cc1N N1(C(c2c(C)nc(C)s2)=O)CCC2C1CCN2C(c1ccc(F)c(Br)c1)=O N1(C(CC(CN(C)C)O)=O)CCOCC(CNC(c2cn(CC3CC3)nn2)=O)C1 c1(C(=O)NC2C(CC)N(C(c3ccsc3)=O)CC2)nn(C)c(C(F)(F)F)c1Cl N1(c2cc(NCC3(CCOC)CC3)nc(COC)n2)CC2CS(=O)(=O)CC2(C)C1 Cc1cc(C)n(CCNC(C2C(O)CCN2C(=O)CNC(C2CC2C)=O)=O)n1 Cc1ccc(C(N2CCOC(CN(C)C(C3CCCC(C)(C)C3)=O)C2)=O)nc1C C1(NC(c2cc(CO)[nH]n2)=O)CCN(C(=O)CN2CC(CF)C2)C1 c1(CCC)cccc(NC(=O)C(CC)N(C(=O)C(CN(C)C)CC)C)c1 N1(C(CCCCC)=O)C(CNC(C2(CN(C)C)CCCCC2)=O)CC2COCC12 C1(C(N2CCC(NC(CCCc3nc(C)sc3)=O)C2)=O)CC2C=CCC(C1)C2 N1(C(C2CC(C)CN2C(c2ccc(N3CCCC3)nc2)=O)=O)CC2C(C1)C2(F)F N1(C(=O)CCCCF)CC2CN(C(=O)C(F)C3CCOC3)CC2C1 C(CCCCC(=O)N1CCC(CC)C1C(=O)NCC(C)C#N)OCC C(C1CCc2ccccc21)N(C(=NCc1ccc(C)s1)NCc1ccco1)C c1(C(=O)NC(CCOC)C(=O)N2CCC(COC)C2)cc2n(n1)CCC2 Nc1ccc(C(N2CCC3C(NC(C4C=CCC4)=O)C23)=O)cc1F C1(NC(C(C(C)O)C)=O)CC2(C1)CC1(CC(NC(=O)Cc3ccc(Cl)nc3)C1)C2 N1(C(C(C(C)(C)C)CNC(c2cc(CO)on2)=O)=O)CC2(C1)CC1(CCC1)C2 c1(C(C)C)cc(C(=O)NC2CC(N(C)C(C3CC4(CCC4)C3)=O)C2)n(C)n1 Cc1ccc(-c2cn(C3(C(=O)O)CC3)nn2)c(C(=O)N(c2cccc(I)n2)C)c1 C1(CC(=O)N(C)CC2(NC(c3nc(C(C)C)oc3)=O)CC2)CC2COCC12 C1(NC(c2[nH]c(=N)sc2)=O)CCC(CNC(C2(C(=O)N(C)C)CC2)=O)CC1 C1(C(=O)Nc2nnc(C)n2C)CC(F)CN(Cc2cscc2Br)C1 C1(SC)CCN(N(CC2CC2)CC2CC2)CC1 C#Cc1ccc(C(N2CC3CC3(C(=O)Nc3c(C)cccc3F)C2)=O)cc1 c1(C(N(C)CC2CCCN2C(c2cnc(C3CC3)s2)=O)=O)ccc(N)cc1[N+](=O)[O-] NC1CC2(C1)CC1(CC(C(=O)N(C3CCCCC3)CCO)C1)C2 C1(CC(C)(C)C)CN(C(=O)CCC2CCC(=O)C2)CCN1C(=O)CSC1CC1 C1(C(=O)OC)C(=O)NCCN1C(c1cc(F)ccc1C)C(=O)NCCCSC c1(C(N2CCOC(c3cn(Cc4ccccc4Cl)nn3)C2)=O)cccc(F)c1F C1(C(=O)NCC#C)CC2(CC2)CN1C(=O)C(C)NC(N)=O c1(CCC(=O)NC(CNC(CC2(N(C)C)CC2)=O)(C)C2CC2)cccnc1 c1(OC)cc2cc(c1O)CCN1CC3CCN(C3C1)C2=O.C1(N(C)C)CC(O)C1 C(=O)(N=c1[nH]c(Cl)cnc1Br)C1C(NCc2c(OC)ncc(Br)c2)C1 CCC(O)C(=O)NCCC(C)N(C(=O)COCC(=O)NCc1ccccc1)C C(CC1=CCCCC1)NC(C1CN(C(c2cccc(O)n2)=O)CC1F)=O c1(NC2C(C(F)(F)F)CCN(Cc3n[nH]c(C)c3C)C2)c(F)cccc1[N+](=O)[O-] C1(C(N(C(CC)C)C)=O)CN(C(c2cn(CC)cn2)=O)CCC1(C)C Cc1nc(C)n(CC(=O)N(C2CC(NC(=O)C=Cc3ccoc3)C2)C)n1 c1(OCCOC)ccc(Cl)cc1C(=O)NC1CN(C(c2n[nH]cc2C)=O)CC1O c1(C(=O)NC(CN(C(=O)C(C2CCC2)OC)CC)C)cc[nH]c(=N)c1 CC1OCCN(C(c2cc[nH]n2)=O)C1C(N1CCCN(C(N)=O)CC1)=O C(=O)(C(C)(C)S(C)(=O)=O)NCC1N(C(CCc2c(OC)cccc2)=O)CCCC1 O=S(=O)(c1ccc(N2CC3CC3C2)cc1Cl)NCc1cccc(F)c1 N1(C(COc2cccc(C)c2)=O)CC(NC(c2cc(=N)[nH]c(Cl)n2)=O)C2(CC2)C1 CC1(C(=O)Nc2cc(F)ncc2F)CCCN(C(c2c(Br)cccc2Br)=O)C1 c1(C(N(CCN(C(=O)CCC=C(C)C)CC)CC)=O)nnc2ccccn12 C(=O)(CC(C(=O)NC1(C(=O)NCC2CCOCC2)CCCCC1)NC(C)=O)OC c1(CCC)nc(C)c(C(=O)NC(C2CCCC2)CNC(c2c[nH]c(Br)c2)=O)o1 N1(C(c2cnc(C)nc2C)=O)CCC(NC(C2(C)CC2)=O)CC(C)(C)C1 C1(NC(CCc2c(C)n[nH]c2C)=O)C2CC1CN(C(c1ccc(=O)n(C)c1)=O)C2 N(C(=NCC1CCCO1)NCC1CCC(C)CC1)C(C#C)CCC N1(C(C2N(C(C(c3ccn(C)c3)C)=O)CC(F)C2)=O)CC(O)C(N=[N+]=[N-])C1 C1(CCC)CN(C(c2c(C)cccc2O)=O)CCN1C(=O)C(C1CCCC1)OC Cc1cc(C(=O)NCCC(C)NC(C2(CO)CCCO2)=O)sc1C Cc1nn(C)c(C)c1C1OCCC1NC(C1CC2(C1)CC(CNC(=O)C(C)C)C2)=O C(c1cnccn1)=CC(=O)NCC(CNC(C(F)=C(C)C)=O)(C)O Cc1cc(=NC2CN(C)Cc3ccccc32)[nH]c(=NCCOc2cccnc2)[nH]1 CC1CCCN(CCc2nc(CCc3cccn3C)n(-c3cccnc3)n2)C1 C1(C(=O)NCC2(CN(C)C(c3csc(O)n3)=O)CC2)CCCC2(CCOC2)O1 c1(C(=O)NC2C(CNC(C(C)NC(C3CCC3)=O)=O)C2)cnncc1O N1(C(C2CC=C(C)CC2)=O)CCN(C(=O)CC(O)c2ccccc2)C(C)C1 N1(C(CSCC=C)=O)CCCCC(CNC(=O)C(C)N2CC(C)C2)C1 CN1CCN(C(c2ccc(COC(C)(C)C)c(F)c2)C(=O)NCC(F)F)C2CC12 c1(C(NOCC(=O)NC(C)CCC2CCCC2)=O)ccccc1 c1(C(c2cn(C3CCC(C(=O)NCCCC(=C)O)C3)nn2)=O)cc(Cl)c(Cl)n1C C12C3CN(CC13)C2=O.C1(CC(=O)OC)CCCN1C(C1CCCCC1)=O C1(O)(CNC(=O)N(C2CC2)Cc2ccccc2)CCN(N2CC(O)C(F)C2)C1 C(C)(C(C)(C)NC(c1cnc(Br)s1)=O)NC(CCNC(C)=O)=O O=C(N=c1[nH]ncs1)NC(CCc1ccccc1)C(F)(F)F N1(C(CC(C(C)C)C)=O)CC2CCC1CC2NC(=O)Cn1cnnc1O N1(C(COCCOCC)=O)CCN(C(=O)Cc2cc(Cl)ccc2Cl)CC1COC CN(C1CCc2ccccc2C1)N1CC(C)(C)C1C1CCN(C(=O)C2CC2)CC1 c1(CC(C)C)cc(C(=O)NCC2CCN2C(=O)CSC2CCOC2=O)n(C)n1 N1(C(c2cc(CCC)ncc2)=O)CCCC2CN(C(=O)Cc3cncs3)CCC12 C(=O)(C(C)(C)C(N)=O)NCC(CC(=O)N(C)CCN(C)C1CC1)C1CCC1 C1(N(C(C2C(=C)CC2)=O)C)CCC(NC(c2ccncc2N)=O)CC1 c1(C(N(C2CCN(C(CC3(C(=C)F)CCC3)=O)C2)C)=O)nc[nH]c2ncnc1-2 N1(C(CCn2cc(-c3cnc(C)s3)nn2)=O)CCC(CSc2cccs2)CCC1 c1(OC)ccc(C(=O)NCCN(C(C2OCCOC2C)=O)C2CC2)nc1Cl CC12CN(C(c3cnc(O)s3)=O)CC1CN(C(c1ncccc1N(C)C)=O)C2 C(=O)(CCCCC(C)CC)N1CC(O)(CNC(COCCSC)=O)C1 N1(C(C)(C)C)CC(C(N2CCC3C(NC(=O)CCCn4cncn4)C23)=O)CC1=O c1(C(N2CCCC(CC(=O)NC3(CF)CCC3)C2)=O)cccn2nccc12 c1(C(N2CCOCC(CNC(C(C)NC(=O)NC)=O)C2)=O)ccccc1S(C)=O CC1(C(=O)NC2CCC2NC(c2ccc(F)s2)=O)CC=CC1 c1(C(=O)NC(CCCCNC(CC(=C)C)=O)C)cc(OC)ccc1F CC(C)CC(CNC(=O)CCCOC(C)C)C(=O)NCC(C)(F)C(C)C C1(CNC(C2(CC)CCCCC2)=O)(NC(=O)C(N)=O)CCC(F)(F)CC1 CCC(C(=O)NCC1=CCN(C(C2(c3ccccc3)CC2)=O)CC1)C(C)(C)CC C1(CCC(=O)NC2CC(C)(NC(c3cc(C4(C)CC4)n[nH]3)=O)C2)CCCCN1C c1(CN2CCOCC(NC(c3ccoc3)=O)C2)n[nH]c2cc(Br)ccc12 Cc1cc(C#N)cc(NC(C2CCCOC2)C)n1 CC1(NC(C23CC(SC(C)(C)C)(OC2)C3)=O)CCCN(C(=O)C(O)P(C)(C)=O)C1 C(=O)(CC(C)(C)SC)N(C1CCN(C(C2CCC=CO2)=O)C1)CC C(=O)(C1=CCCC1)NC(C(=O)NCCCC(=C)Cl)C1CCCO1 N1(C(CCS(=O)(=O)N(C)C)=O)CCC(C)(C)C(NC(c2cc(F)cnc2Cl)=O)C1 C(CO)(C(C)(C)CO)NC(C1N(C(c2[nH]cc(C(C)=O)c2)=O)C(C2CC2)CC1)=O O=C1CCC(CC(N2CC3CC2(CNC(=O)C(O)Cc2ccccn2)C3)=O)CC1 c1(C(=O)NC2CCN(C(C3CC(=C)C3)=O)CC2O)ccc(Br)c(C)c1C C(C(C(=O)NCCCCc1cnc[nH]1)NC(=O)COC1CCN(C(C)=O)C1)OC C1(C)(C(N(C(C(=O)OCC)C)C)=O)C2CC3CC(C2)CC1C3 Cc1cccc(C(=O)NCC(O)CN(C(=O)C(C)(C)CN(C)C)C)c1F CC1(NC(=O)Cc2csc(Cl)n2)CC(NC(C2CC2Cl)=O)C1 Cc1cc(N(C2(C)CC=CC2)C)ncc1S(=O)(=O)NC1CC(C(F)F)C1 CCC(CC)C(F)C(=O)NCCOCCC(=O)NCC1CCN(C(N)=O)C1 CCC(C)CC(C(=O)NC(C)C(=O)N(CC)CC)NC(=O)C(O)CCC(C)C C1(NC(COCC=C)=O)CCC2(CCCN(C(c3cocc3Br)=O)C2)C1 N1(CCC(=O)N(CC(c2ccccn2)O)C)C(=O)C2CC=CCC2C1=O C#CCCC(N)C(=O)N1CC(C(=O)NOC)CC1(C)C Cc1ccc2cccnc2c1C(=O)NCCC(C)(C)NC(=O)CC1CCCC1C C(=O)(C1CCc2ccc(OC)cc21)NCCCN(C(C1C(=C)C1)=O)C Cc1ccnc(F)c1-c1cnc(CNC(c2cc(O)ccc2F)=O)nc1 C1(C(N(CC)CC2CC2)=O)N(C(C2CCC(O)CC2)=O)CC12CCCC2 c1(C(CO)NCc2n(C(C)(C)C)ncc2)ccc(N2CCCCC2=O)cc1 C1(C(=O)NC(CCOC)CNC(C2(C)CCOC2)=O)CC2(CCCC2)C1 C(CC(C)C)(C(=O)Nc1ccc(SC)cc1)NC(C=CC(CC)C)=O C1(CCC)CN(C(=O)C=CC=C(Cl)Cl)CCN1C(=O)CC1CCCC(C)(C)C1 c1(C(N(C2CN(C(C3CCC(CCC)O3)=O)C2)CC)=O)ccc(OC)nn1 CC1C(NC(c2cc(C3CC3)nn2C)=O)CCN1C(c1ccc(C2CC2)cn1)=O C1(NC(c2cc(OC)cc(Cl)c2)=O)CC2(CCN(C(C3CCC3(C)C)=O)C2)C1 C1(NC(C=NOC)=O)CN(C(C2(c3cccc(C)c3)CC2)=O)CC1(C)C CC(CC(=O)NC1CN(C(c2cc(F)c(O)c(F)c2)=O)CC1(C)C)C(C)(C)C c1(C(=O)NC(C)CCNC(c2ccc(Cl)cc2C(F)F)=O)ccc2ccnn2c1 N1(CC=C)CCN(C(c2nc(C(=O)Nc3ncccc3SC)cs2)=O)CC1 Cc1ccc(Br)c(F)c1C(=O)NC1(C)CCOC1C1CC1 C#Cc1ccc(C(=O)NC(CN(C)C(C2(CC(F)(F)F)CC2)=O)CC)c(F)c1 N1(C(c2cnc(C3CC3C)s2)C(=O)NCCCC(=O)OC)CCNC(=O)C1(C)C C1(C(N2CSCC2C(=O)NCC(C)C(F)F)=O)(OC)CCC(C)C1 c1(N2CCCC(C(C)NC(c3c(C)c(I)ccc3)=O)C2)ncnc2cc(I)sc12 c1(C(N2CC(NC(CCC#C)=O)C(C=C)C2)=O)cc(Br)ccc1[N+](=O)[O-] c1(OC)cnc(F)c(C(=O)NCC2(OC)CN(C(C3CCCN(CC)C3)=O)C2)c1 c1(CC(=O)N(CC)CC2CCN(C(=O)CCN3CCC3)CC2)cccc(C)c1Cl c1(OC)ncc(CN2CCCC(NC(c3nccnc3C(N)=O)=O)CC2)cc1C N1(C(c2c(C)cc(C)o2)=O)CCCC(O)(CNC(C2CC(C3CCC3)C2)=O)CC1 N(C(=NCc1ccccc1)N1CCC(C(=O)Nc2cc(C)ccn2)C1)C(C=C)C c1(C(N(C(CNC(CCCNC(C)=O)=O)C)C)=O)ccc2ncnc(O)c2c1 C(CCC(C(=O)NC1CCOC1)N1CCC(CF)CC1)=C(C)C CCCC(CCC)C(=O)NC1CCC(N(C)C(c2onc(Br)c2C)=O)C1 c1(CC)cc(C(F)(F)C(N2CC(OC)CC2COC(=O)OC(C)(C)C)=O)n(C)n1 CC12COCC1CN(C(C1N(C(=O)C3=NNC(=O)C3)CC13CCCC3)=O)C2 c1(C(=O)NCCC(C)N(C)C(C2CNC(=O)N2)=O)ccc2c(n1)CCC2=O CC(C)C(O)CC(=O)NC(Cc1ccoc1)C(=O)N(C)CCC1CN(C)C1 Cc1cc(OCC(N2CCC3(C2)CN(C(=O)C(C)C)C3)=O)c(C(C)C)cc1Cl c1(C(N2CC(C(=O)NCC34CCCN3CCC4)NCC2)=O)cc([N+](=O)[O-])ccc1F N1(C(c2c(C)nn[nH]2)=O)CCC(C)N(C(c2cc(Cl)cnc2O)=O)CC1 C(=O)(C(CCN(C)C)N(C)C)NCCC1N(C(C(=C(C)C2CC2)F)=O)CCC1 C(C(O)C(=O)N(CC(=O)NCCN1CCCC1)C)N(C)C c1(C(N(CCC)CCNC(=O)CC2COCCN2C)=O)cc(F)c(CO)c(F)c1 Cc1ccc(C(=O)NC2CC3CCC2N3C(=O)C(O)C(C)C)cc1C C#Cc1ccc(NC(=O)C(=O)Nc2cnn(CN3CCCCC3)c2)cn1 C(=O)(C1=CCC2CCC1N2C(C1(C)CCC(F)(F)CC1)=O)OC(C)(C)C N1(C(C=CSC)=O)CC(NC(=O)C(CC(C)C)NC(=O)OC(C)C)CC12CCC2 N12CCC(C)(CC1)C2.C1(C(C)(C)C)CC=CC(n2cc(C3C4COCC34)nn2)C1 Cc1cc(C(N2CC(C(C)NC(C3COCCO3)=O)C2)=O)cc(Cl)n1 N1(C(CCN(C(C2CC2C(F)F)=O)CCO)=O)CC(F)(F)C1 c1(NCCC2CCC(NC(c3n(C)nnc3)=O)C2)ccccc1[N+](=O)[O-] CCC(C)(C(c1nnnn1C1CCCCC1)NCCCc1ccco1)OC c1(C2(NC3(c4nnnn4C)CC(OCC)C3)CC2)cccc(Cl)c1 C1(C(=O)NCCN2CC(OCC)C2)C=CCN1C(=O)CCn1cnc(=N)[nH]1 N1(C(=O)CNc2nccs2)C2CCC1CC(NC(C1(O)CCOC1)=O)C2 c1(CC2CC(CNC(C3CC(OC)C3)=O)C2)csc(CC(c2ccccc2)=O)n1 N1(C(c2ccncc2)C(=O)Nc2cccc(CC)c2)CCCC(C)C1C(=O)OC N1(C(C(=O)Nc2cc(C(C)(C)C)no2)=O)CCOCC1C1CC(F)(F)C1 c1(C(N2C(CNC(C3C(C)C3C)=O)CC2)=O)nccc2[nH]ccc12 C1(CC=C)(NC(=O)Cn2nnc(-c3ccsc3)n2)CN(C(=O)CC2CC2(Cl)Cl)C1 c1(C(C)=O)cccc(CCn2cc(CC3CN(C(=O)CCC(F)F)C3)nn2)c1 c1(C(C(=O)Nc2cc(C(=O)N(CC)CC)c(Cl)cc2)O)cc(F)c(F)c(F)c1 C(=O)(C#CC1CCCC1)N(C1CCC(NC(c2c(OC)c(Cl)sc2)=O)CC1)C c1(N(C)Cc2ccn(CC)c2)ccc(OC)c(OC)c1 n1(CC(=O)NC(C)(CNC(c2nccnc2O)=O)C2CC2)cnc([N+](=O)[O-])n1 C(c1ccc(F)cc1F)=CC(=O)NCC1CC(NC(C2(O)CCSC2)=O)C(O)C1 c1(C(=O)OCC)cn(CCC(=O)N2CC(c3nnc(OC)s3)C2)nn1 CC1CCN(C(C2CC(CNS(C)(=O)=O)C2)=O)CCN1C(=O)Cc1cccnc1 C(=O)(C(C)CCCC(C)=O)NC(CCC)C(N1CC(O)CC1(CC)CC)=O c1(C(C(=O)NCC2C(NC(c3ccn(CC)n3)=O)C2)N(C)C)c(F)cccc1Cl c1(C(C(=O)NCCN(C)C(C23CCCC2C3(F)F)=O)(C)C)ccc(F)c(Cl)c1F C(CCS(C)=O)(C(=O)NC1CCC(NC(c2ocnc2C2CC2)=O)CC1)N(C)C C1(CNC(CSC)=O)CC(C(C)C)CCN1C(c1cnccc1Br)=O Cc1ccc(F)cc1C(N1CCCCC(NC(=O)C(C)(O)Cc2ccccc2)C1)=O N1(C(CC2(OC)CC2)=O)CCCCC1CNC(=O)Cn1cc(C)c(C(F)(F)F)n1 c1(C(=O)OC)ccc(C=CC(N2CCCC2CN(C)C(C2CC2C(C)C)=O)=O)o1 C1(CNC(c2c(F)ncc(C)c2)=O)CC2(CCC2)CN1C(c1ccnc(Cl)c1)=O N1(C(c2cc3n[nH]c(C)c3cc2)=O)CCCC(C2CN(C(c3cnc[nH]3)=O)C2)C1 c1(C(N2C(CC(=O)OC)COCC2)=O)cncn(C)c1=O.CC(CO)n1cccn1 C1(N(C(=O)Cc2ncc(C)s2)CC)CCN(C(C2CC2F)=O)CC1 C1(C)(C(=O)NC(CC(=O)NC)C)CCN(C(C2CC2(F)F)=O)CC1 Nc1c(C(=O)NCCC2CCN(C(=O)C#CC3CC3)C2)cc(Cl)cc1Cl CC1=C(C(=O)NCC2CCOC2C(=O)NCC2CC2c2ccco2)CC1 c1(C(N2CC3C(N(C(CC4CCCC(C)O4)=O)C)C3C2)=O)c[nH]c2nccc-2c1 N1(C(CC(=O)NCC#C)=O)CCN(C(C2(c3ccc(F)cc3)CC2)=O)CC(O)C1 N1(C(C2CC(C)(CC)C2)=O)CCC(NC(c2ccc(SC(C)C)cc2)=O)C1(C)C C1(C(=O)NC(CC(=O)OC)C2CC2)C(C)CCN1C(c1cncc(NC)n1)=O CCC(O)C(F)(F)C(=O)NC1CC(NC(=O)CN2CC(C)(C)C2)C(O)C1 C1(C)(CNC(c2cnc(CC)nc2O)=O)CC(F)(F)CN1C(c1cn(C)cn1)=O CN=C(NCc1cnc(C)cc1C)N1CCCC(OCCOC)C1 c1(C(C(=O)NCC(CC=C)NC(=O)COCCCF)OC)ccccc1Cl C(=O)(CC(C)(C)O)NCC1(C(N)=O)CN(C(c2c(CCC)[nH]cc2)=O)C1 N1(C(C=CCN(C(=O)CC2CCSC2)C)=O)CCN2CCCCC1C2 c1(CCC(=O)NC(C2CN(C(C3(C#N)CC3)=O)CCO2)C)cc(F)ccc1F C1(NC(c2c(C)nc(COC)s2)=O)CC(F)CN(C(c2cc(C)ncc2C)=O)C1 C=CCC(CNC(c1[nH]ccc1C1CC1)=O)C(=O)N1CCC(CC)C1 C12(C(=O)NCC(C(C)(C)O)F)CCN(C(C3(N(C)C)CC3)=O)CCC1C2 CN(CCCC(=O)NC(c1ccc(F)cc1)CNC(=O)Cn1cncn1)N=O c1(C(C)C)cc(C(=O)NCC2CCCCN2C(=O)Cc2cncs2)ccc1F C1(NC(=O)CC2(O)CCCCC2)CCCN(C(=O)CCc2ccsc2)CC1F C12CCCCCC1C(=O)N2.Cc1ccc(C(N2CCCC2C2(C)CC2)=O)s1 CCC(CC(=O)N(CC(C)NC(=O)C(C)=C(C)C)C)NC(N)=O c1(C(=O)NC2CCCC(NC(CC=CC)=O)C2)cc(C)c(Br)c(Cl)c1 C1(CCC)(NC(=O)COCC)CCN(C(=O)C(C(C)(C)C)NC(N)=O)CC1 C(=O)(C1Cc2ccccc21)N1CCN(C(c2cc(CSCC)on2)=O)CC1CC N1(C(C2CC(C#C)(O)C2)=O)CC2CC1CCN2C(c1cccc(C2CC2)c1)=O C1(NC(CCc2c(C)nn(C)c2)=O)CCN(C(C2CNC(=O)O2)=O)CCC1CO Cc1ccnn1CC(=O)NC(CNC(=O)C(C)Cc1ccccc1)C1CC1 C(=O)(C(F)CC(C)(C)NC(C1CCCSC1C)=O)Nc1cn(CCC#C)nc1 CCCCC(C(=O)NC(CCN(C)C(C1CCCC2CC12)=O)C(C)C)NC(N)=O c1(CC)cccc2c(C(=O)NC3CCCCC3NC(C3CCCCS3)=O)c[nH]c12 N1(C(CCC=CCC=C)=O)CCC2(CCCN2C(=O)C(C)CC=CC)C1 c1(C(=O)NCC2CC(OC)CN2C(C2COCCOC2)=O)cc(O)ccc1Cl c1(COC(C)C)cc(C(=O)NC(C)C(C)NC(=O)Cc2ncc(Cl)s2)ccc1F c1(CC(=O)NCCC(C)NC(CCn2ccc(C)n2)=O)nn(C)cc1[N+](=O)[O-] c1(C(=O)NCC(C)CN(C(=O)CCC2CC2)C)n[nH]c2c1CCCC2 C1(CC)CN(C(c2cccc(C3(O)COC3)c2)=O)CCN1C(c1ccc(C)o1)=O C(=O)(C(C(C)C)C(C)C)NC1C2CN(C(c3ccc(C(CC)C)cc3)=O)C1CC2 C1(C(=O)NCC2(NC(c3cc(F)c[nH]3)=O)CCC2)CSC(c2ncccc2O)=N1 CC(CC(C)(C)CO)NC(=O)CC1N(C(c2nc(Cl)cs2)=O)CCC1(C)C C#CCC(CC(F)F)C(=O)N1CC(NC(=O)C2=C(C)CCC2)C2CCCCC12 O=C(C1=C(c2ccccc2)CCCC1)NC1CC(NC(c2ccsc2Cl)=O)C1 C(=O)(C(C(C)(F)F)c1ccccc1)NCCN(C(=O)C=CC(=O)NC1CC1)CC C1(C(N(CCCOCCNC(=O)CSc2nc[nH]n2)C)=O)CC12CC(O)C2 c1(C(=O)NC(c2cc(Br)c(F)cc2F)C)cc(F)c(N)c(F)c1 N1(C(=O)CC2CC=CCC2)CC2CCCC2(Nc2ncncc2Cl)C1 N1(C(C(c2cccc(C)c2)C)=O)CC(=O)NC2CN(C(c3cnsn3)=O)CCC12 c1(OC)cc(C)c(Cl)cc1C(N1CCN(C(c2cc(F)c(C)c(F)c2)=O)CC1)=O N=c1[nH]cc2c(c1C(N1CCC3(CCC3NC(=O)C3=CCSC3)CC1)=O)CCC2 N1(C(Cc2nnc(C)o2)=O)CC2(C)CN(C(C3CC3C)=O)CC2(C)C1 C(=O)(C(C)(C#N)CC(=O)OC)NCCNC(CCCOCCOC)=O.C1CCS1 Cc1onc(Cl)c1C(=O)NC1CN(C(C2SCCCS2)=O)CC1CC1CC1 CC(C(=O)NC(C)CSC(C)(C)C)OC1CCCC1 C1(NC(=O)Cn2cncn2)CN(C(c2cnn(C3CCC3)c2)=O)C2(CCOC2)C1 c1(CC(=O)NCC2(C)CCN(C(=O)CN3CC=CC3)C2)cccc2ccccc12 c1(CCC(=O)NCC(C(C)(C)C)NC(C(COCC)C)=O)cc(F)cc(F)c1 C12(C(=O)NC3C(CNC(C4N(C)CCCC4)=O)COC3)CCC(CO)(CC1)C2 C1(NC(CCn2ncc(C)c2)=O)C2CCCN(c3ncnc(O)c3Br)C2C1(C)C N1(C(c2cc(C)n(C)n2)=O)CC2CCC1C(CNC(=O)C(C(C)(C)C)N(C)C)C2 c1(C(N2C(C)(C(N3CCC(C(=O)OC)C3)=O)CCC2)=O)ccc(F)cc1C c1(C2CC(=O)NC2)cccc(NC(C2CCC(C(N3CCCC3)=O)O2)=O)c1 c1(C(=O)NCC2CCCCN2C(=O)CC2CCCO2)cc2nccc(Cl)c2s1 c1(NC(c2cncc(-c3ccc(C#C)cc3)n2)=O)cnc(Cl)c(C#N)c1 C(C(C)C(C)C(=O)N(C)CC1(NC(c2ncoc2C2CCC2)=O)CC1)OC C(=O)(C1=COCCO1)NCC1CC(N(C)C(c2sccc2OC(F)F)=O)C1 CCC(CC)(CCNC(=O)CCc1cncnc1)NC(c1nccc(N)c1Cl)=O C(C)(C(O)C(=O)NCCCCNC(=O)CCc1cccc(N(C)C)c1)SC C1(C(=O)O)(NC(c2ccc(CC(C)C)s2)=O)CC2(C1)CC1(CC(F)(F)C1)C2 C#CC(C(C)OC)NC(C1(C)CC(NC(c2cc(O)cs2)=O)C1)=O N1(C(C(CC)C)=O)CC2CCN(C(=O)CC3CCC(O)C3)C2C1C c1(C(=O)NCCC(=O)NC(CN(C(C(C)C)=O)C)(C)C)ccccc1 c1(C(=O)NCC(CNC(=O)CC#N)OC)cnc(S)n1C1CC1 CC(F)(F)C(F)C(=O)NCC1CC(C(=O)NCC2CCC(O)CC2)=NO1 c1(C(=O)NC2CCN(Cc3ccc(C#C)s3)CC2O)c[nH]c2cc(OC)ccc12 N1(C(C2C(C)(C)CCO2)=O)CC2(C1)CN(C(c1ccc(-c3ccccc3)s1)=O)C2 N1(C(c2nc(COC)sc2)=O)CCCC(NC(C2(C)CCCS2)=O)CCC1 c1(N(C)CCO)ccc(C(c2nnnn2C)NCC2C(C)(C)C2(C)C)nn1 N1(C(CS(=O)(=O)NC)=O)CCCC12CCN(C(=O)Cc1ccc(O)cc1C)CC2 C1(C(N(C(C(=O)NC(c2ccccn2)C)C2CC2)C)=O)CC(N=[N+]=[N-])C1 c1(CN2C(C(=O)NC3CN4CCC3CC4)CC3CC32)c[nH]c2cccc(Cl)c12 C(CCC(C)(C)C(=O)NCCOC(C)(C)C)N(C(CC1CC1)C(=O)O)C c1(CC(=O)NCC(Cn2cc(CC3CCNC3=O)nn2)OC)ccc(Cl)c(Cl)c1 N1(C(C=CCC(C)(C)NC(=O)Cn2[nH]cnc2=N)=O)CCCC2(C=CCO2)C1 C=CCC(CC(=O)NCc1cnc(CC)s1)NC(=O)C(O)C1CC1 C1(CNC(C(CO)N(C)C)=O)CC2(CCC2)CN1C(c1cc(O)nc(O)c1)=O C1(NC(C2N(C(C)C)CCCC2)=O)CC12CCN(C(=O)CCP(C)(C)=O)CC2 c1(NCc2ccc(C(C)NC(C3(C=C)CCC3)=O)cc2)nccc2ncncc12 C(C)(C)(CCC(=O)NC(C)CC(C)C(F)F)NC(c1cccc(CC)n1)=O N1(C(C(C)OCCCC)=O)CCN(C)C(C(=O)NCC2(C3CC3)CCCO2)C1 C(C)(CNC(c1c(C)ccnc1C)=O)(CC(C)C)NC(CCN(CCC)C)=O c1(CN(c2c(C)nn(C)c2C)C2CC3CNC2C3)ccc2oc3ccccc3c2c1 c1(C(=O)NCC2CCCN(C(C3(C#N)CCOC3)=O)CC2)nccc2cc[nH]c12 c1(CNC(C2(C)CCN2Cc2ccnc(N3CCCC3)c2)=O)c(F)cncc1Br Cc1ccc(=N)[nH]c1C(=O)NCCOCCNC(C1CC=CCC1C(F)(F)F)=O c1(CC)cnoc1C(=O)NC(C)CCCNC(=O)C=Cc1ccsc1 C1(C(=O)NCCCN(C)C(C2CC3(C2)CC3F)=O)(C(N)=O)CCCCC1 C1(CNC(C=C(C)Cl)=O)CN(C(C23CC2COC3(C)C)=O)CC12CC2 C1(O)(C(=O)NC2C(NC(C3CC3C(F)(F)F)=O)CCOC2)CCOCC1 C1(NC(C=CC(N)=O)=O)CCCN(C(=O)CCC2CCOC2)C1 Cc1cc(CO)oc1C(=O)N(C)CC1CCN(C(=O)CC2COCCN2C)C1 N1(C(CC(CC)O)=O)CCC2(CCCN2C(c2cc(CO)oc2C)=O)C1 N1(C(CC2(CSC)CC2)=O)CC(OC)CC(NC(=O)CC2C=CCCC2)C1 C(=O)(C(C)C(F)(F)F)NC(C)CCCNC(C1(C(C)(F)F)CC1)=O C12(C(=O)NCC3(CO)C(C)(C)C3)CCC(CN(C(C34CC(C#N)(C3)C4)=O)C1)C2 O=C(C1CSc2ccccc21)NC1(CCNC(C2(C(F)(F)F)CC(O)C2)=O)CC1 C1(C(=O)NCC=C(C(=O)NC(CCC)CO)C)(CO)CC(C)(C)C1 C1(C(=O)NCc2ccc(C(=O)OC)s2)CC=CCC1SC(CO)C(=O)O c1(C(=O)NC(CNC(C(C(C)C)O)=O)C(C)(C)C)nc2ncc(Br)cc2[nH]1 C1(NC(c2c(C#C)cnn2C)=O)CN(C(C2COC(=O)N2)=O)CCC1(C)C S(=O)(=O)(CC(=O)NCCC1CCN(C(=O)Cc2ccccc2C(N)=O)C1)NC c1(NC(C23CC(CO2)C3)CNC(c2n(CC)nc(C3CC3)c2)=O)ccc(C)cc1Cl c1(C(=O)NCC2N(C(C3N(CC)CC3)=O)CC2)cc(N)cnc1C c1(NC(CC(=O)N2CC(CNC(COC(C)=O)=O)C2)=O)cccc2ccccc12 CCCCCCCCS(=O)(=O)N1CCCC1CS(N)(=O)=O O=C1CCN(C(c2ncccn2)=O)C(C(N2CC=CC(O)C2)=O)C1 CC1CCOCC1C(=O)NC1CN(C(C2(c3cccc(F)c3)CCCC2)=O)C1 C1(CC#C)(C(=O)NCCN(C(=O)CC23COC(C)(C2)C3)CC2CC2)CC=CCC1 C1(CNC(c2cc3c[nH]nc3s2)=O)CCCCN(C(C2CC23CC(F)(F)C3)=O)C1 N1(C(c2nncc(CCC)c2)=O)CCN(C(=O)C(C(CC)CC)OC)CC12CC2 CC1C(NC(=O)C(C)(C)N2CCCC2)CCCN1C(c1cc(C2CCC2)[nH]n1)=O CC(C(C)C(=O)NCC12CC(NC(=O)C(C)O)(CO1)C2)C(C)(C)C C1(C(=O)NC23CC(NC(=O)COc4cccc(F)n4)(C2)C3)CCC2CC2C1 N1(C(C2(C)CCCNC2=O)=O)CC2CCC(C1)N2C(c1cccc(N)c1O)=O N1(c2cc(COC)ncn2)CCC(CNC(C2CCCSC2)=O)C(C)C1 c1(C(=O)NC(C(C)C)C(C)NC(C2C3CCC2CC3)=O)ccc2ccoc2c1 Cn1ccc(C(=O)NC(c2ccccc2)CNC(=O)CC2(C)CC2(Cl)Cl)cc1=O c1(-c2nc(C)c(N(C)C)s2)cc(C(N2CCCC(CO)(CO)C2)=O)c2c(c1)CCO2 N1(C(c2cnc(C(=O)O)o2)=O)CCOCC1CCc1ccccc1 C1(NC(CCCOCC)=O)CN(C(C2(COC)CC=CC2)=O)CC1C c1(C(=O)NC(C(C)C)CCNC(=O)CCS(C)(=O)=O)cc2c(cc1N)OCCO2 CC(O)C(C(N)=O)NC(=O)C(CN(C)C)NC(=O)CC1CNC(=O)O1 c1(C(=O)NC2C(NC(C3C(C(N)=O)C3)=O)CCC2)cccc(C(F)(F)F)c1 C(N=c1nc(N2CCc3nc(Br)sc3C2)c2[nH]ccc2[nH]1)C1CC(OCC)C1 CCC(C)CC(C)C(=O)N1CC2CC1(c1cn(C3CCCCC3)nn1)CO2 N1(C(c2c(CC)ccs2)=O)C2CCC1CN(CC(N1CCCCC1=O)(C)C)CC2 CCCC(O)C(CO)NC(=O)CCN(CCCO)C(=O)CC1CCCCC1 N1(C(C2CSCCN2C(c2cnccn2)=O)=O)C2CCC1COC2 c1(C(N2C3CN(C(CC(C(C)C)C)=O)C(C3)C2)=O)ccc2cncn2c1 C1(CCNC(CN(C)C2CC2)=O)CCCCN1C(C1CCCCC1O)=O Cc1ccnnc1C(=O)NCCC1CN(C(=O)Cc2nonc2C)CC1C N1(C(c2n(CC)nnc2)=O)CC(C(=O)NCC2(C)CCOCC2)C2(CCC2)C1 S(=O)(=O)(c1cnn2ccc(NC3CCn4nccc4C3)nc12)NC(C)(C)C C(CSC)(C(=O)NC(C)CC1CN(C(=O)C(c2ccccn2)O)C1)OC C(=O)(C1=C(F)CN(C(C2CNC(=O)C2)=O)CC1)NC1C(C#N)CCCC1 N1(C(COC(C)=O)=O)CCC(C)(CNC(c2ccc(C(F)(F)F)nc2)=O)CC1 C1(C(=O)NCC2CC(NC(c3cc(C)c(F)nc3)=O)C2)CCc2nn[nH]c2C1 N1(C(C(CC(C)C)OC)=O)CC2(C=C(C(=O)NC3CC(=O)N(C4CC4)C3)CO2)C1 C1(C(=O)NC(CO)(CO)CO)CN(C(=O)C(c2cccnc2)O)CC1F c1(C(=O)NCC2CC(NC(C3C(C)(C)OC3(C)C)=O)C2)cc2n(n1)CCCC2 C1(C)(NC(CCCn2c(C)ncc2)=O)CCCN(C(=O)CC(=O)N(C)C)C1 c1(C(C)=O)ccccc1C(=O)NC1CCCC1NC(=O)C(C)(C)c1cnco1 n1(CC)nc(C)c(CNC(N2CC(Cc3ccccc3)C2)=O)c1C c12cc(c(Br)cn1)C(=O)N2.c1(COC)cccc(C(N2CCOCC2)=O)c1 C(CC(C(=O)NC(CNC(c1sccc1C(F)F)=O)CO)OC)OC CC1CC(C(=O)NCC(Cl)Cl)CN(C(=O)CNC(=O)OC(N)=O)C1 N1(C(c2ccc(NC(C)C)nc2)=O)CCC2(C1)CN(C(c1ccncc1F)=O)C2 CC1(C)COCCC1C(N1CCC(=CCNC(C2CC3(C2)CC3(F)F)=O)CC1)=O c1(C(N2CC(CC(C)NC(=O)CSc3n[nH]c(=N)s3)C2)=O)n[nH]c2c1COCC2 CCC(CC)(CC)C(=O)N1CCC(C)(NC(c2ccc3nc[nH]c3n2)=O)C1 N1(C(=O)OCC)CCN(C(=O)Cc2cnccc2C)C(CC(F)F)C1 C1(O)(CNC(c2cc(CNC(C(C)NC=O)=O)sc2)=O)CCOC1C N1(C(C2CCN(C(c3n[nH]c(C)c3Br)=O)CC2)=O)CC(C)NC(=O)C12CC2 C(C(C)C(F)C(=O)NOC(C)CC)NC(c1c(CC)n(C)nc1)=O OCC(CO)(CO)CCCNC1CCN2CCC1C2 CC1CN(C(=O)C(O)c2ccsc2)CC1CNC(=O)CCCOc1ccccc1 C1(NC(C=CC(C)C)=O)CCN(C(=O)CCC2CCC(=O)N2)C12CC2 C1(NC(Cc2cc(C)c(F)cc2)=O)CC2CC(NC(=O)CC3(C)CC3)CC2C1 Cc1cccnc1CC(=O)NCC(C)NC(=O)C(C)n1cccn1 c1(OC)cccc(C(C)C(N2CCCC2CN(C(=O)C(C)OCC(C)C)C)=O)c1 c1(OC)ccc(N2CC(C(=O)OCC=CCNC(=O)CC3CC3)CC2=O)cc1 C1(OC)CS(=O)(=O)CC1NCc1cnn(CCc2ccccc2)c1 c1(OC)ccnc(C(=O)NC2(C)CCN(C(C3CCCS(=O)(=O)C3)=O)C2)c1C c1(CNC(C)C(=O)OCCN2CC(C(N)=O)C2)ccccc1 C1(NC(=O)C=CC2CCOCC2)CCCCN(C(C2CCCC2C2CC2)=O)C1 N1(C(c2ccccn2)=O)CCCCC(NC(c2cn(CC(=O)OCC)nn2)=O)C1 C1(C)(C(=O)NCCCN(C)C(C2(C3CCCO3)CCOCC2)=O)CCCCO1 CC1CC(=Cc2ccc(Cl)cc2F)C(=O)c2ccccc21 N1(CC(=O)NCC2CC2CNC(c2ccc[nH]2)=O)CSCC1=O N1(C(C(CC=C)C)=O)CCC2(CC1)CC(NC(=O)CCNC(=O)COC)CCO2 C#CCC(CC(=O)NCc1nc(CC)cs1)NC(=O)CNC(C1CC1C)=O c1(C(N2CCN(Cc3n(C(C)C)ccn3)CC2)=O)nccc2ccncc12 C1(C(N(CCN)C)=O)CCC(c2cccc(C(F)(F)F)c2)CC1 C1(C)(CC)CC(C(=O)NCCCCCCNC(=O)C(C)CN(C)C)CCO1 N1(C(C2(C#N)CC3CCC2C3)=O)C2CCCC1CC(N)C2 C1(OCC(=O)NC(C(C)N(C(C2(SC)CSC2)=O)CC)C)CCN(C)CC1 c1(CNC(NC2C(C)C2)=NCCNCCS(C)(=O)=O)cc(CO)n2c1COCC2 N1(C(CN(C2CC2)CC)=O)CC2CC2(CNC(=O)CCCc2nccs2)C1 c1(N2CC(Cc3ccccc3)OCC2)nccc(=NCC2C3CCC(F)(F)C23)[nH]1 c1(C(N(CCCCNC(C(CC)SC)=O)C)=O)ccc2c(c1)CCCN2C(C)=O C1(C(=O)NC23CC(CNC(C4(CC)CC4)=O)(C2)C3)CC(OC)C(OC)C1 c1(NC(N2CCC(c3ccccc3)C2)=S)cccc2ccccc12 N1(C(c2cnn(CCCC)c2C)=O)CCC(CNC(C2(CC)CCC2)=O)C(C)C1 N1(C(C=CCOC)=O)CC2(CC(NC(c3snnc3C)=O)C2)C1 C#Cc1ccccc1CN1CC(CC(C)C)C1 c1(CC2CCN(Cc3n[nH]c(C)c3C)C2)nc(O)c2cc(Cl)ccc2n1 CC(CN=c1nc(N2CCC3(CC=CCO3)CC2)c2cccc(F)c2[nH]1)C(F)F N1(C(C(C)C)=O)CCC2(CCCC2NC(=O)CCCn2ccnc2)C1 c1(C(N2C(CCNC(c3cncc(N)c3)=O)CCCC2)=O)cccc(=S)n1O N1(C(c2ccc(N)cc2F)=O)CCC(NC(=O)CC2=CCCC2)C(CO)CC1 [N-]=[N+]=NC1(C(N2CC3CC2CC3O)=O)CCN(C(=O)Cc2ccoc2)C1 c1(N(C23CC(N)(C2)C3)Cc2c(OC)cccc2Cl)ncc2cc(Br)cnc2n1 Cc1nnc(N2CCC(c3cccc(F)c3)C2)nc1C.C1(=O)NNC(=O)CN1C NS(=O)(=O)CC(=O)NCCC1CCCN(C(c2cncc(O)c2)=O)C1 N1(C(C2CC(NC(c3c(OC)ccnc3)=O)C2)=O)CCC2(CCNC2=O)CC1 CCCC(C(=O)NCC(C)(CC(C)C)NC(c1sc(C)nc1C)=O)C(C)C Cc1sc2ccccc2c1CNC(c1cccc(-c2cnc3cncn3c2)c1)=O CCC(C)CCC(=O)N1CC(CNC(c2cccnc2N)=O)C(C)(C)C1 c1(CC)cc(C(=O)NC2CCCN(C(C3CC4(OC)CC3C4)=O)CC2)c(C)nn1 C(c1cn[nH]c1)=C(C)C(=O)N1CCC1C(=O)NC(C)COC(F)(F)F C(=O)(CC(C)(C)C(F)(F)F)OCc1c(OCC=C)cccc1 C1(C(=O)OCC)C(C2CC2)CCN1C(=O)Nc1cc(OC(C)(C)C)cnc1F N1(C(c2ccc(SC)o2)=O)CC(CNC(=O)C(C)(O)C2CCC2)C(F)(F)C1 c1(C(N2CC(N(C(=O)CN3C(=O)C=CC3=O)C)C2)=O)ccc(F)nc1N(C)C C1(NC(CCOC)=O)CCN(Cc2ccccc2-c2cnco2)CC1(C)C C1(NC(COC(CC)(C)C)=O)CN(C(c2n[nH]c(CCCC)n2)=O)CCC1(C)C C1(CNC(C2CN(C(N(C)C)=O)C2)=O)(CNC(C2CC(O)CN2)=O)CC1(F)F c1(C(=O)NC(C)C#N)cc2c(s1)CCN(Cc1ccc(Br)c(Cl)c1Cl)C2 C1(O)(CNC(=O)C(O)c2cnc[nH]2)CC(NC(=O)CCOC2CC2)C1 C1(C(=O)NCCCCC2CN(C(C(C)(C)F)=O)C2)C2Cc3ccccc3C12 C(=O)(C(C)CC=Cc1ccccc1)NCC(N(C(CSCCOC)=O)C)C1CC1 C(C(CNC(=O)Cc1nc([N+](=O)[O-])n[nH]1)C(F)(F)F)NC(c1cncc(C)n1)=O C1(C(CNC(C=C(C)Cl)=O)F)CCN(C(c2cc(C(F)(F)F)on2)=O)CC1 C1(C)(CNC(CC(CN(C)C)O)=O)CN(C(C2CCCCC2)=O)CCO1 C1(CC(=O)NCC(CNC(C(c2c(OC)cccc2)O)=O)C)CC(=O)NC(=O)C1 C(=O)(CCCC(=O)N1CSCC1C(=O)NCC1CCCC1N(C)C)OCC c1(OCC)ccc(C(=O)NC2CCN(C(=O)C=C(CC)CC)C2C)cn1 c1(COC(C(C)(N(C)C(=O)OC(C)(C)C)C2CC2)=O)cc(F)c(O)c(F)c1 S(=O)(=O)(c1ccc(Cl)cn1)NC1CC(C(N2CCOC3(CC3)C2)=O)C1 CC1(C)CC(NC(=O)CCCCO)CN1C(=O)COCC1CCCO1 Cc1nc(C)n(C2CCCN(C(=O)Nc3cc(N4CCCC4)ncn3)C2)n1 C=C(C)C1OCCC1C(N1CCC(CO)(CNC(=O)Cc2ccoc2C)CC1)=O CCC(CC(=O)N1CCC(C)CC1C(=O)NCC1CC2(CC2)C(=O)O1)C(F)F N1(C(c2n(CC#C)ccc2)=O)CCCC(CC(=O)N(C2CCCC2C)C)C1 C1(C(=O)NCC2(C)CC(NC(=O)C3=CCCSC3)C2)CCc2ccccc2O1 c1(NCC2(C)CCN(C(=O)CCn3cc([N+](=O)[O-])cn3)C2)ncnc2scnc12 c1(OC)cc(C(=O)NC23CC(CNC(C4(CO)CCCC4)=O)(C2)C3)c(N)cc1F c1(C(=O)NCC2CN(C(Cc3cn(C)nc3)=O)CC2(C)C)nc[nH]c2nccc1-2 C1(OC)CN(C(c2ccc(C(C)=O)cc2)=O)CCC1NC(c1ccc(C)cn1)=O c1(OCC(=O)NCC2CCCN(C(=O)CCn3cccn3)C2)cccc(Cl)c1 CC1(C)CCC(CNC(c2ccc(F)o2)=O)N(C(c2c[nH]c(=N)s2)=O)C1 N1(C(C(C)OCC)=O)CCC(C(N2CC(Cc3ccoc3)C2)=O)C(O)C1 C12(c3nn(-c4ccc(C)c(F)c4)c(-c4coc(Cl)n4)n3)CC3CC(CC(C3)C1)C2 C1(C(CSC)(F)F)CC2CCC(C1)N2C(=O)CNC1CCSC1 c1(CC(=O)NC2CN(C(C(C)C(C)(F)F)=O)C2)cncc2ccccc12 N1(C(C(CCC)NC(N)=O)=O)C2CCC1CC(NC(C1OCC1(C)C)=O)C2 c1(OC)ccc(C#N)c(NC(=O)Cc2csc(=NCc3c(O)cccc3O)[nH]2)c1 CC1(CNC(=O)C(F)(F)CN2CCCC2)CN(C(=O)CCN2CCCC2)CCO1 c1(C2(OC)CC2)cccc(C2CCCN2C(c2cccc(-c3nn[nH]n3)c2)=O)c1 C(=O)(C1CCCc2n[nH]cc21)NCC1N(C(=O)C=Cc2ncc[nH]2)CCN(C)C1 C1(C(=O)NC2CC(CCNC(C(CCC)C)=O)C2)CSc2ccccc2O1 CC(C)(C)C1=NOC(C(N2CC(CNC(c3ccsc3)=O)C3(CCC3)C2)=O)C1 c1(CC(=O)NCCNC(c2nncn2C2CC2)=O)cc(-c2ccco2)on1 N1(C(CCCC(=O)OC)C(=O)NC2CCOC2)CCn2c(nc(C)c2C)C1 CCCC(CCCNC(C1COC1)=O)NC(=O)CCOc1ccc(OC)cc1 C=C(Cl)CC(C(=O)N(C1CC2CCC1O2)C)NC(=O)C(CC)n1cncn1 C12(C(=O)NC(C)(C)CF)CCN(C(c3c[nH]cc3C3CC3)=O)CCC1C2 c1(C(=O)NCC(C)CN(C)C(C2CC3CCC2O3)=O)nn(CC(F)(F)F)cc1Cl C1(N(CC#C)C(C2CCCO2)=O)CCN(C(=O)C(C)SCC2CC2)CC1 CN1CCC2(CCN2C(=O)CC(C(F)(F)F)NC(=O)Cc2cnnn2C)C1 C1(CNC(c2c(C)snn2)=O)CC2(CCN(C(c3cccc(CO)c3)=O)CC2)C1 C1(C(N(CCN(C(C(C)OCC)=O)C)C(C)C)=O)CC(=O)C12CCCC2 CC1CNCCC1CNC(C1CCN(c2ccc(C(F)(F)F)cc2)C1)=O c1(C(N2C(CN(C(=O)CC3(CO)CC3)C)CCCC2)=O)cc2n(n1)C(C)CCC2 C(=O)(C(C)=C(C)C)N(CCCC)CC(=O)NCCNC(=O)OC(C)(C)C C(=O)(C1Cc2ccc(F)cc21)NCC(C)NC(C1CCCN1CC(F)(F)F)=O c1(C(N2CCCC(CC(=O)NC(c3cnc[nH]3)C)C2)=O)cc(Cl)ccc1Cl c1(C(C(=O)OC)N(c2cc(C)ccn2)C(=O)Cc2cccnc2)cccc(C)c1 CCCCCCCCOCC(N1CCN(C(=O)CSc2ccccc2)C(C)C1)=O c1(C(=O)NC2CCC(CNC(c3cc[nH]n3)=O)C2)cc(Cl)c(F)cc1F C1(O)(C(C(=O)NC(C)CC2CCCCC2)NC(CC2C(CC)C2)=O)CCCCC1 c1(SCc2cn(CC3CN(C(C(CO)OC)=O)C3)nn2)cc(C(=O)O)ccc1Cl c1(CC(N2CC3C(CNC(C(C)(C)F)=O)C3C2)=O)cncc2ccccc12 CC1CC(C(=O)NCC(C)(F)CNC(c2cc(C3CC3)no2)=O)CC(=O)N1 c1(-c2c(C(=O)NC3CN(Cc4ccccc4)CC3F)csc2)ccc2c(c1)OCC2 C1(O)(CCNC(C2C(C)C2)=O)CCN(C(=O)CCC(C)C#N)CC1 C#CCC(C)(CNC(=O)COC1CCN(C(c2cnco2)=O)C1)CO CC1CN(C(=O)CC2CCCN2C)CCCN1C(=O)CCCNC(N)=O c1(OC)c(C(=O)N(C(C)CCNC(c2cncc(C(N)=O)c2)=O)C)ccnc1Cl Cc1cnc2c(C(N3CCN(C(C4C5CC6C(C5)C46)=O)CC3CF)=O)cccn12 c1(OC)ccc2c(c1)C(C(=O)N1CCN(C(=O)CC3CCC3)CC1CO)CC2 CN1C(=O)CSC1=CC(=O)N1CCCOC(CNC(C2CC(F)(F)C2(C)C)=O)C1 S(=O)(=O)(c1ccc(N(C)Cc2ccc(Br)s2)c(Br)c1)NCC1(CN(C)C)CC1 C(C)(C1OCCc2sccc21)NC(C(=O)NC(c1c(C)nc(C(C)C)s1)C)=O CCN(OC)C(=O)CNC(=O)C(Cn1cccn1)NC(C1CC(C)(C)CO1)=O c1(C(=O)NC2CCCCC2CNC(c2n[nH]c(O)n2)=O)ccc2nc(Cl)nn2c1 C#CCC(CC#C)C(=O)NC1(C)CC(NC(=O)CN(C)C(C)C)C1 Cc1ccc2c(c1)CN(C(C1CC1NC(c1cnn3cccnc13)=O)=O)CC2 C1(NC(c2c(CC)cno2)=O)CCC(CNC(=O)C(C)CN2CCOCC2)CC1 C1(NC(COCC=C)=O)CN(C(c2cc(-c3cnn(C)c3)on2)=O)CCC1(C)C N1(C(CC2CCC(C)(C)CO2)=O)CCC(CNC(c2csnn2)=O)C(F)(F)C1 Cc1nc2n(n1)CC(C(=O)N(CCNC(c1coc(C#N)c1)=O)C(C)C)CC2 c1(NC(C(C2CCN(C)CC2)NC(C23CC(C2)C3)=O)=O)cn2cc(Cl)ccc2n1 C1(NC(C2CCCCC23CCC3)=O)CCN(C(C2CCSCC2)=O)CCC1CO c1(-c2cn(C(C(C)(C)NC(=O)OC(C)(C)C)C)nn2)ccccc1C(N)=O N1(C(c2c[nH]c(=NC)o2)=O)CCN(C(=O)CC2CC3CCC2O3)C(C)C1 C1(C(N2CC(CCC)C2)=O)CCC(C)(C)N(C(C2CC2Cl)=O)C1 CCC(C)CC(C(=O)NCC(C(C)C)C(C)C)NC(C1CC1Cl)=O c1(C(=O)NCC=CCNC(CC2CCC(C)O2)=O)cccc(C2(C#N)CC2)c1 C1(NC(=O)CCC2CCOCC2)CN(C(c2coc(Cl)c2)=O)C2(CCCCC2)C1 C(CCCCNC(C1OCCO1)=O)N(C(C1N(CC)CC1)=O)C c1(CN2CCC(O)(C(=O)Nc3ccc(Cl)cc3I)C2)c(F)ccc(Cl)c1Br c1(CN2CCC(n3ncc(NC(CCC#C)=O)c3)CC2)cc(C)ccc1[N+](=O)[O-] C1(C(=O)NCC(C(C)(C)C)NC(CC(C)(C)O)=O)CCC(=C(F)F)CC1 C(=O)(C1CCc2nccn21)NC1CCN(C(c2c(SC)cc(Br)cc2)=O)C1 c1(CN(CCC)C)ccc(C(=O)NCC=CCC2(COC(C)=O)CCC2)cc1 C(=O)(C1=CC2CC=CCC12)N(C1CCCCCC1)CC C1(NC(C2N(C(C(CSC)C)=O)CC(=O)NC2)=O)CCC2(CCC2)CC1 C1(C(=O)NCC(C(C)C)O)CC(F)CCN1C(c1cc(O)nc(O)n1)=O c1(C(=O)NCC2CCOC2)[nH]nc2ncc(-c3ccc4nncn4c3)cc12 S(=O)(=O)(c1ccc(C#N)cc1)N1CC2CN(C(c3ccc(CCC)cc3)=O)C2C1 Cc1nn(CC(=O)NC2COCC2CNC(=O)Cc2cncnc2)c(C)c1Cl n1(CCOC)ncc(C(=O)NCC2CCN2C(c2cccc(C(C)C)n2)=O)c1C C(=O)(CC(C)CC(C)C)N(CCC(=O)NC(c1nc(CC)[nH]n1)C)CC c1(C(=O)NCC2CN(C(c3c(C)csc3)=O)CC2C)cccc2nc[nH]c12 C1(CC(=O)NC2CCC(CO)CC2)C=NN(C)C1=O.CC1CNC1=O Cc1ccc(C(=O)N2CCC(C(=O)NC(c3ccccc3)(C)C)O2)cc1C#N C1(C(=O)NC(C)CCNC(=O)CCCc2cnccn2)CCCCN1S(C)(=O)=O N1(C(CC(C)SC)=O)CCC2(CCCN2C(=O)CC2CC(O)C2(C)C)C1 c1(NC(N(C)Cc2cccc(SC)c2)=O)cc(S(N)(=O)=O)ccc1Cl N1(C(=O)OC(C)(C)C)CCC2(CCCC2N2CCCC(CSC3CC3)C2)CC1 c1(C(N2CC(NC(C(C)(C)OC)=O)C(OC)C2)=O)ccnc(C)c1C C1(C(=O)N(C)CCOCCOC)(CC)CCN(C(=O)CN2CCC(=O)CC2)C1 c1(NC(C2C(CNC(=O)CC3C=CCCC3)C2)=O)ccc(O)c(F)c1 N1(c2cc(C)c(Br)cn2)CCCC2(C1)C(=O)NCCN2C N1(C(CC(=O)NC2CC2)=O)CCC2(CO)CN(C(=O)C(F)(F)C3CC3)CC2C1 CCCCC(O)C(=O)N1CCC(N(C(=O)C=C(C)C)C)C(C(N)=O)C1.N1(CC)CCC1 c1(C(C)OC(c2cn(-c3cccc(Cl)c3)cn2)=O)ncccc1Br N1(C(c2ncn(C(C)C)n2)=O)CC(CNC(=O)Cc2cnoc2)OC2(CCC2)C1 C1(N(C(CSCCC)=O)C)CC2CC1N(C(C1CCCC(C)(C)C1)=O)C2 c1(C(C(=O)NCCN(C(=O)CCSC(F)(F)F)C)(C)C)c[nH]c2ccccc12 C1(CNC(c2cc(C)n(C)c2)=O)CCCCCN1C(=O)C(C)C1CCC1 Cc1nn(CC(=O)NC2(C)CC(NC(=O)CS(C)(=O)=O)C2)cc1[N+](=O)[O-] c1(NCCCC(C)NC(c2ccoc2Br)=O)snc(Cl)c1C#N C1(C2(C(=O)NC(=O)CCNC(=O)NOCC(=O)OC(C)(C)C)CC2)CCC(=O)NC1 C(N=c1[nH]c(=NC)[nH]c(=NCc2cccc3c2NC(=O)CO3)[nH]1)C1N(CC)CC1 N1(C(C(C)SCC)=O)CCOC2CN(C(c3csc(C(=O)OCC)n3)=O)CC12 N1(C(Cc2ccc(C)o2)=O)CCN(C(=O)C2=C(Cl)CCOC2)C(C)CC1C c1(N2CCC(NC(C(CCCC)C)=O)C2(C)C)ncnc2c(Br)nn(C)c12 C#Cc1ccc(C(=O)NC(C)C(C)C(=O)NC(C)(CC(C)C)C(N)=O)c(C)c1 C1(C(=O)NC2CCNC2=O)(OC)CCN(C(=O)CC2CCCCO2)CC1 C1(CC(N2CC(C)(CSC)C2)=O)CC(O)CN1C(=O)C(C)O C(=O)(C1=NOC2(CCC2)C1)N(C1CCN(C(c2cn(C3CC3)cn2)=O)C1)CCC CCCC(C(=O)NCCOC(C)C)NC(c1cc(C(C)C)nn1CC)=O C1(C(=O)NC(C(C)NC(=O)Cc2csc(-c3cccs3)n2)C)OCCOC1(C)C c1(C(=O)NC(CNC(C(CCC)C)=O)CC)nn(C(C)C)c(=O)c2ccccc12 c1(OC)cc(F)c(S(=O)(=O)NCC(C)(C)O)cc1Br N1(C(c2n(CC)nc(C)c2)=O)CCC2(C=C(C(=O)NCCSCCO)C2)C1 C1(CNC(c2ccn(C3CC3)n2)=O)COCCN1C(c1cncs1)=O Cc1cc(C(=O)NCC2CCCN2C(=O)COCc2ccnn2C)ccc1F C1(CNC(C(C)OCCOC)=O)CCN(C(=O)CC2CCC(=O)N2C)CC1 N1(C(CN(C(=O)OC(C)(C)C)CC)=O)CCC(CC2CC2)C1.c12nnnn1C2 Cc1nc(C(=O)NC2CCN(C(=O)CCC3(C)CC3)C2C(C)(C)C)cn1C N1(C(C(CC2CC2)NC(CCC2C(C)C2)=O)=O)CCc2n[nH]cc2C1 N1(Cc2cc(C)c(C(F)F)cn2)CC2(COC(=O)N2C)C1 c1(OC)cc(C(N2CC(O)CC2C(=O)N(C(C)C(C)C)C)=O)ncn1 C(C)(C)(CCCNC(c1ccc(-c2cccs2)cn1)=O)NC(CN(C)CC)=O Cc1cc(C(N2CC=CC(NC(=O)C(c3ccncc3C)C)C2)=O)c(C)cn1 c1(C(C)C)cccnc1CC(=O)N(CCCNC(=O)COCCN(C)C)CCO c1(OC)noc(C2CC2)c1C(=O)N(CC(C)CNC(c1ccnc(S)c1)=O)C C=C1CC(C(=O)NC(C(O)CO)C2CC2)(CNC(C2CC=CCC2)=O)C1 N1(C(C2ON=C(C)C2C)=O)CCC(NC(c2scnc2Cl)=O)C(C)(C)C1 C1(CNC(c2c(C)n(C3CC3)cc2)=O)CN(C(C2CC(O)C2)=O)C2CCN1C2 CCCCC(CNC(=O)C=Cc1cnc[nH]1)NC(c1cc(Cl)c(Br)[nH]1)=O Cc1c(C(=O)NCC2CN3CCC2(C)CC3)oc2ccc(Br)cc12 Cc1cc(C(N2CC(NC(c3c(C)noc3C(F)(F)F)=O)C(C)C2)=O)cc(Cl)n1 c1(C(N2CC(C(=O)OC)C2)=O)n[nH]cc1CNC(=O)CC1CC1(C)C C1(C(N2CC=C(C)CC2)=O)CCN(C(c2c(C)noc2N)=O)CC1(C)C C12(C(N3CCC(NC(c4c(C)nncc4)=O)(CF)C3)=O)CCC(O)(CC1)CC2 CC(CS(C)=O)C(=O)NCCCNC(c1cnc(O)c(Cl)c1)=O C1(OC)(OC)CC2(COC(CNC(=NCC3CCOC3)Nc3nccs3)C2)C1 N1(C(C2C(C(C)=O)C2(C)C)=O)CCN(C(C2CCCC3CC23)=O)CC1C c1(OC)cccc(C)c1-c1ccc(CNC(C2CCN(C(C)C)C2=O)=O)nc1 C(=O)(C(F)(F)CCn1cc(-c2ncoc2C)nn1)N1CCC(OCCOC)C1 C1(CNC(C(c2ccn(C)n2)C)=O)(NC(=O)CCC2CCC(=O)C2)CC(F)(F)C1 N1(C(C(C)(C)SC)=O)CC2(C1)C(NC(=O)CC1CCS(=O)(=O)C1)CCS2(=O)=O N1(CC2NCCN(C(C(C(C)C)NC(C)=O)=O)C2)CCC2COCC2C1 C1(NC(C(C)Cc2cnn(C)c2)=O)CC(NC(c2cccnc2Cl)=O)C(O)C1 C=CC(C(=O)N(CCCN(C)C)CCNC(=O)CSCc1cccnc1)OC N1(C(C(C)(C)N2CCCCC2)=O)CCCC(O)(NC(=O)COc2cn[nH]c2)C1 O=C(CCN=c1[nH]ccs1)NC1(CO)CN(C(C2(C(F)F)CCCO2)=O)C1 C1(O)(CN(C(COCC=C)=O)C)CCN(C(=O)CN(C)CCc2ccccc2)C1 C1(NC(C(COCC)C)=O)CCC(NC(=O)Cc2ccc(C(F)(F)F)nc2)CC1 N1(C(C2(C3CC3)CN(C(C3C(C(=O)OCC)C3)=O)C2)=O)CCC2OCCC2C1 N1(C(CCC(N)=O)=O)CCC(C2CC(NC(=O)Cc3ccc4sccc4c3)C2)C1 N1(CC(N2C(CCNC(=O)C=Cc3cnc[nH]3)CCC2)=O)C(=O)CNC1=O C12(C(=O)NC(C)CCNC(=O)CCCCc3ccccc3O)CCC(F)(CC1)C2 N1(C(COCCC)=O)CCC(O)C(NC(=O)C=C2CCC(C)CC2)C1 C(C(C1CCCCC1)NC(=O)C1=CCSC1)(C(C)C)NC(C=C(CCC)C)=O C1(CCC)CN(C(c2cncc(F)c2)=O)CCN1C(c1ccnc(CO)c1)=O C1(CC)C(C(=O)NCc2cc(OC)ncn2)CCCN1C(c1[nH]cc(C)c1C)=O N1(C(CCCn2cc(COC(=N)O)nn2)=O)CCC(F)(C(=O)O)CC1 CN1CC(O)CC1C(=O)NC1CC(NC(=O)Cc2ncc(Cl)s2)C1 C1(CC=C)CCCC1N=c1nc2sccc2c(NCc2nc(C(C)(C)C)cs2)[nH]1 C1(CN(C)C(C2CCC(=O)O2)=O)CCN(C(c2ccnn2CC2CCC2)=O)CC1 c1(C(=O)NCCNC(C2ON=C(CC)C2)=O)ncc2c(F)cccn12 Cc1ccc(C(=O)NC2CC(CNC(=O)COCC3CCOC3)C2)c(Cl)n1 C1(CNC(C2CCCOC2)=O)COCCN(c2cc(O)ncn2)C1 Cc1cc(=NC(=O)C2CC(O)CCN2Cc2ccc(O)c(O)c2)[nH]n1C c1(C(C)C)nn(C)cc1C(=O)NC1COCC1NC(C1(c2cc[nH]n2)CC1)=O c1(C(C2(C)CC2)NC(N2C(CC)CCC2)=O)ccccc1Br N1(C(C(C)OCCC#C)=O)CCC(C2CC2)(NC(=O)COc2cccc(F)c2)C1 CCCCCC(O)C(=O)NC(C1(CNC(c2cn(C)c(=O)c(C)n2)=O)CC1)C c1(OC)ccc(C(=O)NC(C2CN(C(=O)C=Cc3cn(C)nn3)CCO2)C)nc1 N1(C(C#CC2(C)CC2)=O)CCC2C(CCN2C(=O)Cc2nc3c([nH]2)CCCC3)C1 C(=O)(C1CCC(=O)c2cccn21)NC(C1CCN(C(C2CCC(=O)N2)=O)CC1)C c1(C(N2C(CCNC(C(C)CS(C)(=O)=O)=O)CCC2)=O)ccnc2nccnc12 C=CCC(CC(C)C)C(=O)N1CC2CCC(C1)N2C C(=O)(C(C)Cc1ccco1)NC(CC)CNC(=O)CNC(=O)NC c1(-c2cc(CNC(c3n(C)nc(-c4ccccc4)c3)=O)[nH]n2)ccc(F)cc1O c1(C(=O)NC(CCNC(CSCC#C)=O)(C)C)oc(-c2ccccc2)nc1C C12(NC(c3ccsc3C(F)(F)F)=O)CCCC1(F)CN(C(C1CCCOC1)=O)C2 Cc1ncccc1CCC(=O)NCCC(C)(C)CNC(c1ccc(Cl)cn1)=O C(=O)(C(C(C)C)C(C)C)N1CCC(OCCNC(C=Cc2c(C)cccc2)=O)C1 c1(CC)ccc(OCCC(N2CC3CC2C3NC(=O)CCCCN(C)C)=O)cc1 CC(C)CC(C(=O)N1CCCOC(CNC(C2C=CCC2)=O)C1)C(N)=O c1(C(=O)NC(CC2CN(C(C=CC)=O)C2)C)cc(F)c(CO)c(F)c1 c1(C(=O)NCCC2CC(NC(=O)C(Cl)=CCl)C2)c(Cl)ccc2ccncc12 C1(C)(C(=O)NC2(CC=C)CC2)CC(O)CN1C(C1CC(C)(C)CN1C)=O Cc1ccc(NC(C2CCC(O)CN2C(c2cnn(C)c2Cl)=O)=O)c(F)c1F CC1CC(NC(=O)CNC(=O)C2CC2)CN(C(c2occ3c2CCC3)=O)C1 C1(C(=O)NC(CC(C)NC(=O)Cc2ncc(F)cn2)C)C2Cc3ccccc3C12 CON(CCC(=O)Nc1cc(C)cc(O)c1)C(=O)C(C)c1cc[nH]n1 c1(C(N2C(C(=O)NCCCC=C)CC2)=O)cccc2c(O)ncnc12 N1(C(Cc2cn(CC)nc2)=O)CCCN(C(C23CC(N=[N+]=[N-])C2C3)=O)C(C)C1 c1(OCC(=O)N(CCC)CCNC(C2CC2N(C)C)=O)ccc(Cl)c(C)c1 N1(C(c2c(C)ccnc2C)=O)CCC2C(CCCN2C(C2COC(=O)N2C)=O)C1 N1(C(c2c(C)ccc(F)c2)=O)CCc2cc(C(=O)NC(C)C(C)(C)C)ccc2C1 N1(C(C2CC=CC2)=O)CCC(C2CCCN(C(C3CC=CC3)=O)CCC2)CC1 C1(CNC(CC(CN(C)C)O)=O)CC(C(C)(C)C)CN(C(C2(O)CCC2)=O)C1 CC1CCC(CC(=O)NCc2ccc(N3CCCC3)nc2)CC1.C12CN(C1)C2=O N1(C(C23CC(C)C2C3)=O)CC2C(NC(=O)CC3C(C)(C)C3(C)C)C2C1 C1(CNC(CNC=O)=O)(NC(=O)CCc2nnc(C3CCCC3)o2)CCOC1 CC1CC(=O)NCC1C(=O)NCCCOCCCNC(=O)C(C)(F)F C(=O)(C1(C)CC(=O)N(C)c2ccccc21)NC(C(C)C)CCNC(=O)CC(F)F c1(C(N2CC(C)(C(N(C)CCC3OCCO3)=O)C2)=O)cccc(=O)n1O N1(C(C(C(C)(C)C)O)=O)CC(C(N2CC(O)CC2CO)=O)CC12CCC2 C1(C(=O)NC(C)CNC(=O)CCCc2cccs2)CC(C(=O)OC(C)(C)C)=NO1 C=CC1CN(C(c2ccnc(C)c2O)=O)CC1NC(=O)C(C)OCC(C)C c1(OCCCC)ccc(C(=O)NCC2(C)CCCN(C(=O)CSCC)C2)c(Cl)c1 N=c1[nH]c(N2CC(c3ocnc3CNC(=O)CN3CCC3)C2)ncc1[N+](=O)[O-] n1(C(C)C)ccc(C(=O)NC2CN(C(C3CC4(CC4)CO3)=O)CC2(C)C)cc1=O C1(NC(C(C)c2cccs2)=O)CCSC12CN(C(=O)CC1CC3CC3C1)C2 N1(C(CCC(C)OC)=O)CC2(CCCCN2C(=O)CCC=C(C)C)C1 N1(C(=O)NC2CCN(C(CNC(C(C)(C)C)=O)=O)C2)CCc2cccc(Cl)c2C1 N1(C(CCC)=O)CCC(CCC(=O)N(C)CC2(O)CCOC2)C1 C(=O)(N=c1ncc(C#N)c[nH]1)NC(c1ccnn1C)C(=O)OC CC(C)C(C(=O)NCc1ccn(CC(F)F)n1)N(C)C Cc1nc(NC2CCN(C(=O)CSc3ccncc3)C(C)C2)c2ccsc2n1 Cn1cc(CC(=O)NCC2(C)CC(NC(C3(Br)CC3)=O)C2)cn1 C1(C(=O)NCC2CCSCC2)CC(O)CCN1C(=O)C1=C(Cl)CC1 C1(NC(c2c(CC)nc(C)[nH]2)=O)CCC2CCN(C(=O)C(C)n3cccc3)C1C2 C=CCC(C)(C)C(=O)N1CC2(C(=O)NCCc3ccccn3)CC1CO2 c1(C(N2CCC(N(C(C=C(CC)CC)=O)C)C2)=O)ccccc1NCC(F)(F)F CC(=O)CCCCC(=O)N1CCCC1C=CC(=O)N(C)CCO C1(CC(=O)NCC(=CC(=O)N(CC(C)(C)O)CCC)C)CCCCC1 C(C)(C)(CC(C)(C)O)NC(Cn1cc(CNC)nn1)=O N#Cc1c[nH]c2ncnc(N(C3(C#N)CCNC3)Cc3ccc(Cl)c(C#N)c3)c12 C1(CNC(c2csc3nnsc23)=O)(NC(C2CCO2)=O)CCC(F)(F)CC1 c1(OCC)cc(C(=O)NCCCC(C)NC(=O)CC2COCCO2)cc(F)c1 c1(C(=O)NCC(C)(CNC(=O)C(F)C2CCOC2)OC)cc(C)ccc1O c1(C(N2CCCC2Cc2ccncc2)C(=O)NCC)cc2cc(C)ccc2s1 c1(C(N2CCC(CN(C(c3scc(OC)c3)=O)C)C2)=O)cc(C2CC2)nn1C C(=O)(CCCCN=[N+]=[N-])NC(C)(CNC(=O)Cc1cnc(C2CC2)[nH]1)CO CC(CNC(=O)CN(C(=O)CCC1(C)CC1)CC1CC1)CC1CCC1 N1(C(c2n(C)c(=O)ccc2)=O)CCCC2(CCN(C(=O)CC3CSCCS3)C2)C1 Cc1ccc2occ(CC(=O)NC3CC3CNC(=O)Cc3sc(O)nc3O)c2c1 C#CCCC(O)C(=O)NCC1(C(N)=O)CN(C(=O)CCCN=[N+]=[N-])C1 c1(C(=O)NC(CCCNC(c2ccn(CC(C)C)n2)=O)C)csc(S(N)(=O)=O)c1 Cc1c(O)ccc(C(=O)NCC2(CN(C)C(C3(C)CC4CCC3C4)=O)CC2)c1C c1(C(=O)NC2CCCC(C(=O)NC(CC=C)CC)C2)nnc(O)nc1O N1(C(CC(C)CF)=O)CC2(CCN(C(c3ccnn3CCN(C)C)=O)CC2)C1 C(=O)(C(CCC)C(=O)OC)N(C(C)C(=O)NC1CCC(C2CC2)CC1)CCC C(CC(C)C(=O)N1CC2CC2C1CNC(=O)CCNC(=O)C(C)(C)C)OC N1(C2C(C)(C)CCNC2)CCC(C2(O)CC2)CC1 C(=O)(C(CC1CCCCC1)N1CCC(n2cccn2)C1)NC(C)C C12(C(N3CCN(C(C(C(=O)OCC)(C)C)=O)CC3)=O)CCCCC(=O)N1CCC2 C12(C(N3CC(C#N)C3)=O)CC(CN(C(=O)C=Cc3ccsc3)C1)C2 CCC(CC)(CN=c1[nH]c(C(C)C)nc(C)c1Br)NC(c1cccc(OC)n1)=O N1(c2nccc(C)n2)CCOC2(CCN(C(=O)CCC3CC3(C)C)CC2)C1 C(C)(CCN(C(=O)CCC1CC1(Cl)Cl)C1CC1)OC CC1(NC(=O)CN2C(=O)CNC2=O)CCC(NC(C2(Cl)CC23CCC3)=O)CC1 N1(C(C)=O)CCC(C(=O)Nc2ccc(C(C)Sc3ccccc3F)s2)C(C)C1 c1(C(=O)NC(CCNC(c2c(C)n(C)cc2)=O)C)cnc2ccccc2c1 C1(O)(CN(C(=O)CC2(O)CCCC2)C)CCCN(C(=O)C(F)n2ccnc2)C1 CC1CCN(C(=O)COCc2ccccc2)CCN1C(c1ncncc1Cl)=O N1(c2nccc(OC)n2)CCN(C(c2cc(C(F)(F)F)[nH]c2C)=O)CC1C C(C(=O)NCc1nc(C(=O)NCC2CCCCCC2)co1)(C(C)C)OCC Cc1c(C(=O)Nc2cccc(F)c2C(=O)NC2CCC(=O)NC2=O)ccc(Br)c1F C1(C(C)C(=O)N(C)CCOCCN(C(=O)CCOC2CC2)C)CCCOCC1 C#CC1(C(N2CC(CN(C(=O)C(C)(C)OC)C)C2)=O)CCCC1 Cc1cncc(C)c1C(=O)NCC1CCN(C(=O)CCCc2cccnc2)CC1 c1(-c2ccc(C(=O)NNC(=O)C3CCC3)cc2)ccc2cncn2c1 C1(C(C)NC(c2cccnn2)=O)CCCC(NC(c2cc(C3CC3)nn2C)=O)C1 c1(N(C)C)cccc(C(=O)NCC2CCCCN2C(c2ncc[nH]2)=O)n1 c1(OC)cc(F)cc(C(=O)NCCNC(c2sc(F)cc2Br)=O)c1N C(=O)(CS(=O)(=O)CNC(=O)C(CO)NC(=O)C(F)(F)F)NC1C(C(C)C)CCC1 C1(CC)CCCN(S(=O)(=O)N2CCC(CN(c3ncc(C)s3)C)C2)C1 CC(C)(C)CC(=O)NNC(=O)NC1CCCCC1S(C)(=O)=O c1(CN(c2n(CCC=C)c(-c3cccc(Cl)c3)nn2)C)cc(F)ccc1Br c1(C2N(C(C3CNCCC3CO)=O)CCC2)ccc(Br)cc1F Nc1cc(C(N2CC=C(CNC(=O)CC(F)(F)F)CC2)=O)ncc1F CC1CN(C)C(=O)CN1N1CCC2(CC1)CN(C(=O)OC(C)(C)C)C2 CC(C)CCC(C(=O)NC1CC12CCOCC2)NC(c1cnn(C(C)C)c1)=O c1(OCCCOC(C2CC(C)SCC2)=O)cccc2cccnc12 c1(OC)cc(OC)nc(N(C2CNCC(F)(F)C2)C(=O)CCSC)n1 C=CC1(CC(=O)N(CCN(C(=O)Cc2cc(Cl)n(C)n2)CC)CC)CCCCC1 c1(OC)cnn(C)c1CNC(c1nncs1)C C1(CN(C(=O)C=Cc2ccn(C)c2)C)CN(C(=O)C(O)CC(N)=O)CC12CC2 c1(OC)cc(C(=O)NCC2CCC2NC(=O)Cc2c[nH]nc2O)sc1S(N)(=O)=O c1(C(=O)NCc2c(C3CN(C(c4n(C)ncc4)=O)C3)ocn2)cc2ccncc2[nH]1 c1(OC)ccccc1CC(=O)NCC(O)CNC(c1oncc1C)=O c1(C(N2CCC(OCCNC(CCCCN(C)C)=O)C2)=O)ccnc(Cl)c1Cl C1(C(C)C)CC(C(=O)OCCN2CC3(COC3)C2)CCO1 N1(C(CN(C(CC(CC)C)=O)CC)=O)CCOC(C)CC1 N1(C(C2CN(CCC)C(=O)C2)=O)CCCC(C)(CNC(c2nnc(C)s2)=O)C1 N1(C(=O)C=CC2CCCC2)CCCCC1C1CCCN1c1nc2ccccc2o1 Cc1cc(CCC(=O)NC(C)CCCNC(C2(C)CCCC2C)=O)nn1C C(=O)(CCC(F)(F)F)NC(c1ccccc1)CNC(=O)CCC1CCCOC1 c1(CN2C(C(=O)NCc3ccc(NC(C)=O)cc3)CC(F)C2)cc(Cl)cnc1Cl C1(C(C)C)(C(=O)NCC2CC(C)(C)CO2)CCCN1C(=O)CC1(O)CCOCC1 c1(NCC(=O)NCC(CNC(=O)C=CCO)O)ccccc1Br C1(C(=O)NCC(=O)N(CC)CC)C=CCN(C(C23C=CC(CC2)C3)=O)C1 C(F)(C(=O)N1CCC(C(=O)NC2CC23CCCCCC3)O1)=CCC CS(=O)C1(CNC(=O)COC2CCN(C(c3cscc3Cl)=O)C2)CC1 c1(C(N(C(C)CNC(C2(C)CC(C)(C)C2)=O)C)=O)ncn2c1CCC2 CON1CCC(C(=O)NCCC2CCCN(C(=O)Cn3cccc3)CC2)CC1 n1(CC(=O)NC2CN(C(CSCCC(C)C)=O)CC2O)ncn2cccc2c1=O N1(CC(N2CCC(C)(NC(C)=O)C2)=O)Cc2ccccc2OC1=O CCC(CC)C(C)C(=O)NC(C1(O)CN(C(=O)Cc2cccc(C)c2Br)C1)C C(CC(C(=O)NCc1nncn1C)NC(C1CC2CCC2C1)=O)OC CC1CN(C(c2cc(Cl)c(Br)cn2)C(=O)NCCC2CC2)Cc2c[nH]nc21 C(c1cncnc1O)=CC(=O)NC1(C2N(C(c3c(C)scn3)=O)CCC2)CC1 Cc1nccn1CCC(=O)NCC1CCC(NC(=O)C(C)CO)C1 N1(C(C=CC(C)NC(C(C(=O)OC)(C)F)=O)=O)CC2(CCC(O)CC2)C1 C1(C)(NC(CSCCC)=O)CCN(C(C23CCC(OC)C2C3)=O)C1 C(=O)(C(C(C)Sc1ccc(C2(C(F)(F)F)N=N2)cc1)C(C)C)OCC c1(C(=O)OC)cc(CNC(=O)NC2CCC(N(C)C)C2)ccc1C C1(CC(=O)NCC2(CNC(C(C)NC(=O)NC)=O)CCC2)COCCO1 C(=O)(C1=CNC2=NCCCC2=C1)NCC1C(C)CN(C(=O)CSc2cn[nH]c2)C1 C1(CC)CN(C(=NCCF)NCCc2ccc(OC)nc2)CC(C)S1(=O)=O Cc1c(C(=O)NCC2CCCC2NC(C2(N(C)C)CC2)=O)cc(C(C)(C)C)n1C c1(CCC(=O)NC2CC(O)(CNC(C(C)=C3CCCC3)=O)C2)ccc(F)c(F)c1 c1(CC(N2CCC(CNC(C3CCC(OC)CC3)=O)C2)=O)ccc(F)c(Cl)c1F C1(c2ccccc2)(CNCCCCCOCC)CC2(CC2)C1 c1(C(=O)NC2CN(C(c3cc(C4C(C)C4)on3)=O)C2)c(F)ccc(Cl)c1N N1(n2c(-c3n(CCOC)ccc3)ncc2)CCC(C(=O)OCC(C)=O)C1C1CC1 C(=O)(N1OC2CCC1CC2)C1(F)CCN(C(c2ccnc(O)c2)=O)C1 c1(C(=O)NC2CN(C(c3c(Cl)cn(C)n3)=O)CC2(C)C)cc(F)c(F)cc1Cl C(=O)(C#CC1(C)COC1)NC1CCC(C)N(C(=O)C(O)Cc2cnc[nH]2)C1 N1(C(C=CCCC)=O)Cc2ccccc2C(NC(=O)Cn2nnc(=O)[nH]2)C1 CC(CC(=O)NCc1ccc(CCNC(=O)Cc2cc[nH]c(=N)c2)cc1)C(F)F c1(C(C)C)cc(C(=O)NC2CCC2CNC(c2cnn(C)c2)=O)ns1 C1(C(=O)NC2(C)CN(C(c3cc[nH]c3C3CC3)=O)C2)CCCC(F)(F)C1 C1(NC(c2cccnc2-n2nccn2)=O)CN(C(=O)Cc2cnc[nH]2)C2CC12 C(=O)(C1CCc2nccn21)N1CC2CN(C(c3cc(OC)c(F)cc3)=O)CC2C1 c1(C(N2CCC(C)(C#N)C2)C(=O)NC2COC2)ccc(F)c(F)c1Br N1(Cc2ccc(OC)c(CO)c2)CC2(CCCC2NCc2nnc(C(C)C)o2)C1 C1(C(N2CCC(CC=C)C2)=O)CN(C(C2OCCC2C)=O)CC1(C)C CC1CCC(CC(N2CC(C(C)NC(C34CCCN(CC3)C4)=O)C2)=O)CC1C N1(C(C2C(CCC)CN(C(C3CC=CCC3)=O)C2)=O)CC2CC(C1)N(C)C2 Cc1cccc(C(F)(F)C(=O)NCCC2(O)CN(C(C3NC(=O)C4CC34)=O)C2)c1 C1(C(=O)NC2CCCC2C(=O)NCc2cccc(C)c2Cl)(OC)CCC(C)(C)C1 C(N=c1nc(NC2CCN(C)C2)c2c([nH]1)c(C)nn2C)c1cnn(CCC)c1C N1(C(C2N(CCn3cc(C(C)C)nn3)CC2)=O)CC(N2CCCC2)C(C)C1 c1(OC)cc2c(cc1OC)CCN(C(c1ccc(N3CCCCC3)nc1)=O)CC2 c1(C(N2CCC(NC(C3CCCN(CC)C3)=O)C2C)=O)cc(C)c(C#N)cn1 CCCC(C(=O)NC(C)CN(C)C(C1(NC(C)=O)CCC1)=O)NC(N)=O c1(OC(C)C)ccc(S(=O)(=O)N2CCC(NC(C(CN(C)C)C)=O)CC2)cn1 C1(NC(N(C)C)=O)CCN(C(=O)C(=O)NCC2CC23CC3(F)F)CC1 N1(C(C=CCCC)=O)CCC(C2CCN(C(c3ccnc4[nH]nnc34)=O)C2)C1 c1(C(=O)NCC2N(C(CC(=C)C)=O)CC=C2)cc(-c2ccccc2)oc1C CC1CCCCC1N(C)C(=O)NC1(c2csc(Br)n2)CC1 Cc1cccc(CNC(C2CCN(CC3(C4CCCCO4)CCC3)CC2)=O)c1 c1(C(=O)NCC(CC)NC(=O)C(C)(C)C2(C)CC2(F)F)cccc(Cl)c1N Cc1ccc(C(=O)N(C2CN(C(c3cnnc(O)c3)=O)CC2(C)C)C)cc1Cl C1(Cn2cc(C(=O)O)nn2)CCCCN(C(=O)CCC2CCCCN2)C1 C(C(C)C(F)C(=O)NCCSC(C)C)NC(C(C(C)C)SCC)=O Cn1cc(C(O)CNC(=O)CNc2nc(-c3ccccc3)n[nH]2)cn1 CC1(C)C(C(N2CCC(F)(C(N)=O)C2)=O)CCN1C(=O)CCc1ccsc1 C1(CCNC(c2cccc(CSC)c2)=O)CCN(C(=O)C2=COCC2)CC1(F)F C=CCCC(C)NC(C1(C(C)NC(=O)Cc2sccc2C)CC1)=O C(CC(C(C)C)NC(c1cc(N2CCCCC2)ccn1)=O)N(C(COC)=O)C N1(C(c2cn(CC)nc2)=O)CC(C)N(C(C23CCC(CC2F)C3)=O)C(C)C1 CCCCC(CNC(c1conc1C)=O)NC(=O)OCC.C12CSCN1C2=O N1(C(C2CCCCN(C(C(CC)CC)=O)C2)=O)CCC(C)(C2CC2)C1 N1(C(c2c(SC)ccs2)=O)CCC2C(CCCN2C(=O)CCc2cnccn2)C1 N1(C(c2c(C)nsc2N)=O)CCOCC(NC(=O)C(C)OCCC(C)C)C1 CC(C)CC(CNC(=O)C(c1ccccc1Cl)(C)C)NC(C1(N=[N+]=[N-])CC1)=O Cc1cc2ccc(C(=O)NCC(C)(C)CCNC(=O)CCNC(N)=O)cn2c1 C1(F)(CNC(c2c(COC)ccs2)=O)COCCN(C(=O)CNC(=O)C2CC2)C1 CC1CN2CC1(C)C2=O.C1(NC(=O)CNC(=O)C(F)(F)F)CCC2CC2CC1 C1(O)(C(C)NC(c2cnc(O)s2)=O)CCN(C(C2CCOCC2)=O)CC1 c1(CC(=O)NC(CNC(c2ccc(N(C)C)cn2)=O)CO)cccc2c1OCO2 c1(NC(CCC)=O)cccc(C(=O)NCC2(C)COCCO2)c1 N1(C(c2cc(CC)oc2C)=O)C2CCCC1CC(NC(C1CC(=O)CCO1)=O)C2 c1(C(=O)OC)csc(S(=O)(=O)N2CCC(CC(N)=O)CC2)c1 C(=O)(NN1CC(C(=O)OCC)CC1=O)NCCCC(c1ccccc1)N(CC)CC N1(C(C2CCC3CC2CO3)=O)C(CNC(=O)C(F)(F)C2CC2)CC2CCCCC12 Cc1nc2c(N3CCC(NC(C4CC(C)(C(C)(C)C)C4)=O)C3C)ncnc2s1 C1(CNC(C(C(C)C)NS(C)(=O)=O)=O)C2CCC1CN(C(c1ccon1)=O)C2 CC(C)CCCC(=O)NC(CNC(C1(C)CCC2CC2C1)=O)Cc1ccccc1 N1(C(CC=C(C)C)=O)CCC(N(C(=O)CC(c2ccc(F)cc2)C)CCO)CC1 c1(CC(C)C)cc(C(=O)NCC2(NC(=O)C(C(C)C)NS(C)(=O)=O)CC2)n(C)n1 C1(C(=O)NC(C)(CNC(c2ccsc2C(F)(F)F)=O)C2CC2)CC2OC1C1CC21 Cc1nnc2n1CC(C(=O)NCCCN(C(=O)CC1COC3CC1C3)C1CC1)C2 c1(COC)cc(C(=O)NCCO)ccn1.C12(COC(C)(C)C)CCN1C(=O)O2 c1(SCC(C)C)cccc(C(=O)NCCC(O)CNC(C2(O)CCSC2)=O)c1 c1(C(N2C(c3nnc(NC(C(C(C)C)N(C)C)=O)s3)CCC2)=O)cc2c(s1)CSC2 c1(C(N2CCC(N(CC#C)C(C3CCCC3O)=O)C2)=O)c[nH]c2cc(F)ccc12 c1(OC)ccc(NC(=O)Cc2sc(C3CCC3)nc2C)cc1[N+](=O)[O-] C1(CNC(N(CC(C)(C)O)Cc2ccsc2)=O)CN2CCN1CC2 C1(C(=O)NCCOCCC#C)COCCN(C(=O)CCCCCC)C1 N1(CC2CC(CC(CC)C)C2)C(=O)C2CCC(C3CCCCC3)CN2C1=O C1(C(=O)Nc2cccc(CSC)c2)CCC12CCN(C(=O)COCC(C)C)CC2 N1(C(c2cnc(O)[nH]2)=O)CC2CC1CN2C(c1ccc(C2(O)COC2)cc1)=O C(CC(C(=O)N1CCCC(CC(C)C)C1)NC(C1C(C#N)C1(C)C)=O)OCC C(C(C)C(F)C(=O)NCCc1nc(C)no1)NC(C(CO)OC)=O C#CC1CC(NC(=O)C(C)=CCNC(=O)Cc2ccc(C)s2)C1 c1(NC=O)cccc(NC(=O)C(=O)NCc2cnn(C(F)(F)F)c2)c1.C1CCOC1 C1(C)(CC)CC(NC(C2CC(C)(CC(=O)O)C2)=O)CCO1 N1(C(CC2C(C)(C)C2)=O)CCN(c2nnc(C3CC3)s2)CC1 C1(OCCC)CCN(c2nnc(-c3cc(Br)no3)n2CC)CC1 N1(C(COCC(=C)C)=O)CC(NC(c2cccc(=S)n2O)=O)CCC1C C(C)(CO)(C(=O)NCC1CCCN(C(C2CC(Cl)(Cl)C2)=O)C1)NC(C)=O CC(C)CC(C)CC(=O)NC1CC2(C1)CC2NC(=O)CSc1ccc(Cl)cc1 CC(C)CCC(O)C(=O)NC(Cc1ccc(Cl)cc1Cl)C(=O)N(C(C)CO)C C1(N(C)C(c2cnsc2)=O)CCC(NC(=O)Cc2nc[nH]n2)C1 C1(CC(N)=O)(NC(CC(COC)C)=O)CCN(C(C2CC(OC)C2)=O)CC1 Cc1cc(CNC(=O)C(C)CN(C)C)oc1C(N1CCCCC1CC(C)C)=O c1(CC)nc2c(C(=O)NCCCCCCN(C(=O)C(C)(C)CF)C)ccnc2[nH]1 n1(CC(N2CCN(C(c3ncc(Br)cc3F)=O)C3CC23)=O)ccc2ccccc12 C(=O)(C1=NNC(=O)CC1)NC1(C)CC(NC(c2cn(CC)nc2C(C)(C)C)=O)C1 c1(OC)ccc(CC(N2CCN(C(=O)C=CC3CCCC3)CC2CF)=O)cc1O c1(C(N(C2CCCN(C(=O)NC3CC3)C2)C)=O)ccc(CNC(N)=O)cc1 c1(C(C)=O)cc(C(=O)Nc2nc(C)c(SCCOc3cccnc3)s2)n(C)n1 c1(C(N2CCC(C(C(=O)NC(C(=O)OC)CO)C)CC2)=O)cc(C)cc(O)n1 N1(C(Cn2cc(C(C)=O)nn2)=O)CCCC(CNC(c2nnc(S)n2C)=O)C1 n1(CC(=O)Nc2cc(CC)cc(Br)c2)ccc2ccc(-c3ccoc3)cc12 c1(OC)nscc1C(=O)NCCCN(c1ccccc1)NC(C1CCC1OC)=O Cn1ccnc1-n1cc(CCS(=O)(=O)NCc2nc(O)n[nH]2)nn1 N1(C(C(C2CCCO2)OC)=O)CC(C)(NC(=O)Cc2cc(C)[nH]n2)C1 C1(C(=O)NCCN(CCC)C(=O)OC)CCCN(C(=O)COc2ccccc2)C1 CCCC(C)CC(=O)N1CC(F)CC1CNC(=O)CC1CC1(Cl)Cl C(C(C(F)(F)F)OCC)N(C(C(=C)C)C)Cc1ccccc1 N1(C(C)C(=O)NCc2ccc(C3CC3)cc2F)C(=O)c2ccccc2C1=O c1(CC)nc(=N)[nH]cc1C(=O)NC(C1CCN(C(=O)CCC2CCC(=O)N2)C1)C N1(C(C2(CCC)CCC2)=O)CC2CN(C(=O)CC3CCCS3(=O)=O)CC2(C)C1 C=CCCC(F)(F)C(=O)NCC1(CCNC(C2CN3CCCN2CC3)=O)CC1 C(=O)(C(C)(C)C(O)C(C)C)NC(COC)CC(=O)Nc1ccc(C)nc1 C1(CNC2(c3ccccc3)CN(C(c3ncc(C)cn3)=O)C2)COCCC1(F)F c1(C(N2C(C(=O)NCCCC=C)CSCC2)=O)cccn2cncc12 N1(C(CC(=O)OCC)=O)CCCC2(CCCCN2C(c2ccc(C)o2)=O)C1 CCC(C)(C)C(C(=O)NCc1cccc(NC(=O)COC(C)=O)c1)OC C1(ONC(=O)C2CCCC2)CCCOC1=O.C1(CC(C)(C)OC)CC=CCC1 C1(CC(=O)NCc2c(C(=O)NCCC3CC(C)C3)c[nH]n2)CCCC12CC2 c1(C(=O)NCC(C)(C2CC2)NC(C2C(F)(F)C23CC3)=O)ccc([N+](=O)[O-])cc1N c1(C(N(C(CNC(C(C)NC(C)=O)=O)C)C)=O)ccc(-c2ccnn2C)cc1 C1(CNC(C(C)CO)=O)CCN(C(=O)C(=Cc2cccnc2)F)C12CCC2 N1(C(C2(CC)CCCN2)=O)CCN(C(c2ccccn2)=O)CC1 c1(CC(=O)NC(CC)CN(C)C(C2(c3cccs3)CC2)=O)c[nH]nc1O c1(COC)csc(C(N2CC(CC(C)NC(=O)Cn3cc(C4CC4)cn3)C2)=O)c1 C1(C(=O)NCCC(CC)(F)F)N(C(C2OCCCC2(C)C)=O)CC12CCCC2 N1(C(C2(C)CCC(=O)C2)=O)CCCCC12CC(NC(=O)CN1CCNC(=O)C1)C2 CC(C)C(C)(O)C(=O)NC1CCN(CCOCc2ccccc2)C1 Cc1cc(C(=O)NCCN(C(=O)C(c2cncc(F)c2)C)CC2CC2)ccc1CO N1(C(Cn2cc(CC)nn2)=O)Cc2ccccc2C(NC(=O)Cn2cnnc2)C1 c1(NC)nc(C)nc(N(C)C)c1C.C12CCC(C)(CC1)N2 CC(C)CCCCC(=O)NCC(O)CCNC(c1c(C2CCC2)cnn1C)=O C#CC(C)(C)C(=O)N(CCC(C)NC(c1nc(Cl)c(Cl)s1)=O)C Cn1cc(C(N2CCC(C)(C(F)(F)F)CC2)C(=O)NCCCF)cc1C#N CC1CN(C(=O)CC2CC(C3CC3)C2)CCN(C(c2cocn2)=O)C1 c1(CC(=O)NC(CN(C(=O)C(N)=O)CC)C)csc(C(C)(C)C)n1 Cc1ccc(C(N2CCN(C(=O)C(=O)NCC3CC3)C3CC23)=O)c(N)c1F c1(NC(C(=O)NC(C(C)(C)C)c2ncccn2)=O)ncc(Br)cc1C(N)=O N1(C(CCC(C)OC)=O)CCC2(CCCN2C(c2cc(C)c(Cl)cc2F)=O)C1 c1(C(=O)NC(C(C(=O)OC)O)C)nc2ncccc2cc1C N1(C(C2C(NC(C3C4CCC(F)C34)=O)CCCC2)=O)CCc2cncnc2C1 N1(C(c2c(C)nc(O)s2)=O)CCCC2(NC(=O)CSCC(F)F)CCCC12 C12(CNC(C(C)NC=O)=O)CC(CO1)N(C(=O)C(C)NC(=O)C1CC1)C2 N1(C(CC(C(C)C)O)=O)CC2(C=C(C(=O)NCC3OC(=O)CC3(C)C)CO2)C1 c1(-c2cccc(C)c2)nc(SC23CC(C2)C3)n(C2CCc3c(F)cccc32)n1 c1(CCC(=O)NC(CC)CNC(=O)C=Cc2cscn2)ccc(Cl)nc1 N1(C(C(C)OCC=C)=O)CCC(CNC(=O)CCN2CCC2)(COC)C1 N1(C(CC2(C)CCCC2)=O)CC2CC1CN2C(c1sc(Br)cc1F)=O C(=O)(C(=O)C(C)(C)CC)N1CCN(C2CN(C(CC=CCC)=O)C2)CC1 C1(CCCNC(=O)CO)CCCCN1C(c1cc(-c2ccco2)on1)=O C(=O)(C(F)(F)C(F)F)NC(C1CCN(C(c2c(C)nncc2)=O)CC1)C N1(C(CC(=C)C)=O)CC(O)CC1CNC(C1(Cc2cnn[nH]2)CCCC1)=O c1(C(=O)NC(c2ccc(Cl)cc2)CO)cnc2n[nH]c(-c3ccc(CO)o3)c2c1 N1(C(C2(C(CC)=O)CC2)=O)CCC2CCN(C(C3C=CC3C(=O)OC)=O)C2C1 CC1CCCN(C(=O)C(=O)NC(C)CNC(=O)CSC(C)C)C1 c1(C(N2CCCC(CN(C(C34CC3C4)=O)NC)C2)=O)c(N2CCCC2)cccc1Cl c1(NC(N2CCC(CN(C(C)=O)C)CC2)=O)ccc(S(=O)(=O)C2CC2)cc1 C(c1ccncn1)=CC(=O)NCCCN(C(C)C)C(C1CCCN(C(N)=O)C1)=O C(=O)(C(CC(F)F)c1ccccc1)NCC1N(C(C(C)(C)c2cccs2)=O)CC1 N1(CCN(C(c2sncc2Br)C(=O)NC)Cc2cncs2)CCOCC1 N1(C(CC2CN(C)C2)=O)CCCCC(NC(c2cnc3n2CCS3)=O)C1 c1(SCC(N2CCCC2CCC2CCNC2)=O)ccc(Cl)cc1 C(CCC(C)C(=O)NCC1CCCN(C(=O)C(C)(Cl)Cl)CC1)OC c1(C(N(C2CN(C(=O)CS(C)(=O)=O)CC23CC3)C)=O)cc(=O)c2ccc(Cl)cc2o1 c1(C(N2CCC(N(C(Cc3c(C)nccc3)=O)C)CC2)=O)nnc(Cl)cc1N N1(C(C(CC)(O)c2ccccc2)=O)CCC(NC(=O)CC2C=CCC2)C(F)C1 C1(C)(OCC(=O)NC(C(=O)N(CC(C)C#N)C)C2(O)CCC2)CCCC1 N1(C(c2c(C)ncc(N)c2)=O)C2CCC1CC(CNC(c1c(C)noc1C)=O)C2 N1(C(COCCCCOCC#C)=O)CC2CCC(C1)N2C(C1(C)CCCCO1)=O N#CC1(C(=O)NCCOCCNC(c2cnsc2)=O)CCOC1 Cc1cccc(C(CNC(C2CCN(C)CC2)=O)NC(=O)CCCF)c1 N1(C(C(CCSC)O)=O)CCC(C)(C)C(CNC(=O)C(F)(F)c2ccccn2)C1 C(=O)(CC(=O)N(C(C)(C(=O)NCCCC1CCOC1)C1CC1)C)N(C)C C1(NC(C2(CC#C)CCN(C(=O)COCCCCC)C2)=O)CCN(C)CC1(C)C C(c1cncnc1O)=CC(=O)NCC1(O)CN(C(C2CC2F)=O)C1 c1(C(C)NC2C(C)CN(C(c3cnns3)=O)CC2)ccc(S(C)(=O)=O)cc1 CCC(C)C(C)C(=O)NC1CC(OCC(=O)NCC23CCCC(CO2)C3)C1 C12(C(N(CCCN(C(=O)CCc3cncc(F)c3)C)C)=O)CC(C#N)(C1)C2 c1(C(=O)NC(CNC(CSCC=C)=O)CCCC)cc(S(N)(=O)=O)n(C)c1 c1(C(N2C(CNC(C(CC3CCC3)NC(C)=O)=O)CC2)=O)cc(C)cc(C)c1 c1(NC(c2ncc(-c3cccc(F)c3)s2)=O)ccnc2cc(Br)nn12 C1(C(N2CC(OCC(=O)NC3C(CC)C3)C2)=O)CC12CCCCC2 C1(C(N2CCCC(OCC)C2)=O)CN(C(=O)C(=O)C2CC2)CCC1O c1(C(C(=O)NC(CC)CN(C)C(c2cn(C)c(O)n2)=O)C)ccc(F)c(F)c1 CN1CC2CC1CN2C(=O)C(c1ccccc1)NC(=O)C1=CCCC1 C(=O)(C(F)(F)C(C)O)NC(c1ccccc1)CNC(c1nc(C(C)C)sc1)=O N1(C(C2OCC(C)(C)OC2)=O)CCC2C(CCCN2C(c2cnc[nH]2)=O)C1 c1(C(N(CCNC(C2(C)CNC(=O)C2)=O)CC)=O)ccc(F)c(S(C)(=O)=O)c1 Cc1ccc(Br)c(C(N2CCCC(NC(=O)COc3cccnc3)C2)=O)c1F N1(C(c2ccc(C)nc2)=O)CCN(C(=O)C(F)CC2CCOCC2)CC(C)C1 CC1(C)OCCCC1CNC(=O)CC(O)CNC(C1CCC(=O)O1)=O Cc1ccc(C(=O)NC(C)CNC(=O)CC2CCC(=O)NC2)cc1C#N C1(C(N2CCC(CN(C(CC(C)c3ccccc3)=O)C)C2)=O)COCCN1C(C)=O Cc1cc(Cl)ccc1CC(=O)NCC1CN(C(=O)CCc2ncco2)C(C)(C)C1 c1(CC)cc(C(N2CC(CNC(c3ccc(Cl)nc3N)=O)C(C)C2)=O)ccc1F N1(C(CC=C(C)C)=O)CCC(=CCNC(C23CC(C2)C(C)O3)=O)CC1 N1(C(Cc2c(C)n(C)nc2)=O)CCC(NC(C2(C3CCCO3)CC2)=O)C(F)C1 Cn1nnc2cc(C(=O)NC3COCCC3NC(=O)CCc3ccccc3)ccc12 c1(OC)cc(C(=O)NCC(C)(O)CNC(C2(C)COC(=O)OC2)=O)ccc1F C1(C(N2CCC(N(C(c3coc(C(F)(F)F)c3)=O)CC)C2)=O)CCC(=O)N(C)C1 CC(=O)CC(C)(C)C(=O)NC(C)CC(C)NC(c1c(C)coc1C(C)C)=O N1(C(c2cnn(C)c2F)=O)CCC2C1CCCN2C(c1cc(C(C)(C)C)on1)=O C1(CNC(C2(C)CC(=C)C2)=O)CCCC2(CCN(C(=O)CC(C)C(C)C)CC2)O1 C1(C(N(CC(C(=O)NC)C)C)=O)N(C(c2c[nH][nH]c2=N)=O)CCC1(C)C Cc1c(CC(=O)NC(C)(C)C(C)NC(=O)C=C2CCCCC2)cccc1[N+](=O)[O-] c1(CNC(C(=O)N(C2CC(OC)C23CCC3)C)=O)cn(C)c(=O)nc1O C1(C(N2CC(OCC)(CNC(c3ccc(CO)cc3)=O)C2)=O)CCC12CCCO2 CC1CCC(CC(=O)NCCCCCN(C)C(c2cnn(C)c2)=O)C1 CC(C)CC(C(=O)NC(C(=O)NCC1CC2(CCC2)C1)C1(O)CCC1)C(N)=O C(=O)(C(O)CC(N)=O)N(CC(CN(C(=O)Cc1ccc(SC2CC2)cc1)C)O)C Cc1cc(C(=O)NC2CC2CNC(=O)Cc2cnn(C)c2C)c(F)cc1N N1(C(C(F)=C(C)C)=O)CC2CCN(C(C3CC4(C3)CC(C)C4)=O)C2C1 c1(C(C(=O)NCC(CC=C)NC(C23COCC(C2)C3)=O)CO)ccc(Cl)cc1 c1(C(=O)NCCN(C(CCCCCOCC)=O)C2CC2)cn2cccc(F)c2n1 C1(CNC(COCC(=C)C)=O)CCCC2CN(C(C3C4COCC34)=O)CC12 C(C)(C(C)C(=O)Nn1cnn(C)c1=S)NC(CSCC#C)=O c1(CNC(C(CC)C)C)cc(F)c(N2CCOCC2)c(F)c1 CN1C(=O)c2ccccc2C1C(=O)N(C1CCCC1)CC1(O)CCN(C(=O)CN)C1 N1(C(C2C3(CCN(C(Cc4n(C)ncn4)=O)CC3)C2)=O)CCc2c(cnn2C)C1 Cn1cc2ccc(C(=O)NC34CCN(C(C5(C)CC(F)(F)C5)=O)CC3C4)cc2n1 C1(CC)CCCCC1OCC(N1CC(NC(=O)CSC(C)C)CC1C)=O CCCC(C#N)C(=O)NC1CCCC1NC(c1ccnc(S)c1)=O C(=O)(C(C(C)(C)C)N1CCCC1=O)NCCN(C(C(CC)c1cccnc1)=O)C Cc1cc(C(=O)NCC2(C(=O)N(CC(C)C#N)C)CCCO2)nc(O)n1 c1(C(=O)NC2(CCC)CC2)c[nH]nc1CNC(=O)CC1CC(F)(F)C1 c1(OCC(=O)NCCCC2(NC(CN(C3CCSC3)C)=O)CC2)ccccc1 CCCC(C(=O)NCC(C)NC(C1CCSCC1)=O)S(N)(=O)=O c1(C(=O)OCC)cc(C)nnc1NCC1CCCN1C(c1cc(C)cs1)=O c1(C(N(C2CCN(C(C=C(C)C3CC3)=O)C2)C)=O)cc2ccc(Br)nc2[nH]1 C1(CC)CN(C(=O)C(=Cc2cccs2)C)CCC1NC(C1CC2(CCC2)C1)=O C1(NC(C(C)OCC)=O)CN(c2nc(Cl)nc(C)c2Cl)C2CCCCC12 C1(CNC(c2cc(Cl)n[nH]2)=O)(CO)CCCN(C(=O)COCC2CCCO2)C1 c1(CCC)ccc(C(=O)N(C2CCN(C(C3CC(CC)C3)=O)C2)C)cc1 CCCCCC(C)C(=O)N1CCCC(Nc2cc(COC)ncn2)CC1 C1(NC(Cc2c(Br)cn(C)n2)=O)CC2CCC1N2C(c1c[nH]c(=O)cn1)=O c1(C(=O)NC(CNC(C)Cc2ccco2)=O)ccccc1C(F)(F)F C1(C(N2CCC(CNC(=O)CCc3cnccn3)C2)=O)CCCC(F)C1 C1(=O)C(C(C)CC2CCC2)N(C)CC2CC1C2.c1(SC)ccc(NC(C)=O)cc1 c1(C(=O)NC(C)CCN(C(=O)C(CO)NC(N)=O)C)cc(C(N)=O)cc(F)c1 c1(C(=O)NCC2N(C(c3c(F)cccc3Cl)C)CC2)n[nH]c2c1CCCC2 c1(N(C(c2cc(Cl)ccc2Cl)=O)CC2CCCNC2)ncnc2n[nH]cc12 c1(Cc2nc(C(COc3cccc(OC)c3)=O)sc2)nc2ccc(Cl)cc2s1 C(C(CCN=c1nc(CC(C)C)cc(C)[nH]1)OC)OC C(=O)(C(CC(=C)C)NC(=O)CCCC1CCC1)NC1C(C=C)OCC1 CCC(C#N)C(=O)NCCC1CN(C(c2csc(C3CC3)n2)=O)CCO1 c1(CNC(C(C2N(C(=O)OC(C)(C)C)CCC2)(C)C)=O)ccc2c(Cl)n[nH]c2c1 N1(C(C=C2CCC(C)C2)=O)CC2CCC1C1CN(C(c3cccn3C)=O)CC21 O(P(=O)(CCC1CCN1C(=O)C(=O)NC(N)=O)OCc1ccc(F)c(C)c1)CC CC12CN(C(c3ccsn3)=O)CC1CN(C(c1ccccc1Br)=O)C2 C1(CC(=O)N(C2CC(SC)C2)C)CCN(C(c2nocc2C)=O)C1(C)C N1(C(C2C(CNC(CCCCCN(C)C)=O)OCC2)=O)CC2(CCC1CO)CC2 c1(-c2ccc(NC(=O)Nc3c(C)cc(Cl)cc3Br)cc2)cc([N+](=O)[O-])ccc1Cl C(CCOC)(C(=O)NC1(C(O)CO)CC1)NC(C(CC)=CC)=O C#Cc1ccc(C(=O)NC(CCC)CCCNC(C2CS(=O)(=O)C2)=O)nc1 Cc1c(NC2(c3nnnn3C(C)C)CC3(C(N)=O)CC23)cccc1C#N C(=O)(C(O)CC(F)(F)F)NCC(C)CC(=O)NC1(C)CC(F)C1 C1(CC(=O)NCC(C(C)C)NC(C2(c3cccnc3)CC2)=O)CCC(C)C(C)C1 C1(Cl)(C(=O)NCC(c2ccccc2)N(C(COCCC)=O)C)CC1(C)C Cc1c(C(=O)NC(C)C(C(C)C)NC(=O)Cc2ccsn2)ccn1CCO CCCCC(CC)CC(=O)N(C1CCCN(C(c2csc3cncn23)=O)CC1)C c1(C(N2CCCC(=Cc3ccccc3)C2)=O)ccc2nncn2c1 N1(C(=O)C2=CCOCC2)CCC2C(CCCN2C(C2(O)CCCC2)=O)C1 c1(C(N2CCC(O)C(F)(F)CC2)C(=O)NCC)cccc2cc(OCC)ccc12 N1(CC(CSc2c(OCc3scc(C)c3)cccc2)=O)CC(C)OC(C)C1 Cc1cc(=NCc2ccco2)[nH]c(NC2CCN(CC(F)F)C2)n1 N1(C(c2c(CNC(c3cc(O)cs3)=O)nccc2)=O)CC2(CCC(O)CC2)C1 C1(NC(CCCC(CC)C)=O)CCN(C(c2cnc(S)[nH]2)=O)CC(C)(C)C1 C1(NC(C(C(C)C)NS(C)(=O)=O)=O)CCC2(CC1)CN(C(c1cnnn1C)=O)C2 CC(C)CCCC(=O)N1CC2(Cn3cc(-c4nn(C)cc4Cl)nn3)CC1C2 N1(C(C2CCN(C(C3(CN(C)C)CC3)=O)C2)=O)CCC2CCC(C1)S2 C1(CN(C)C(C2CCS(=O)(=O)N2)=O)CCCN(C(=O)CN2CC(F)(F)C2)C1 C1(CNC(COC)=O)COCCN1C(=O)CNC(=O)Nc1cccc(Br)c1 C1(NC(C(c2ccc(OC)cc2)CC)=O)C2CC1N(C(c1ccncc1F)=O)C2 c1(C(=O)NCC2(OCC)CN(C(=O)C(C)C#N)C2)ccc(NC(C)=O)cc1F C=CC(CC(=O)NCC1CCC1NC(=O)C1=CCSC1)c1ccc(OC)cc1 N1(C(CCC)=O)CCCC(C2(NC(c3n[nH]c(C)c3Br)=O)CC2)C1 S(=O)(=O)(c1ccc(NCCOC2CCC2)c(F)c1)NC(C)C(C)(C)C C1(C)(C(N2CC3(N(C(C4(OC)CCOCC4)=O)CC3)C2)=O)CC(C(C)C)=NO1 C(c1ccccc1Cl)=CC(N1CC(CNC(c2cc(F)ncc2Br)=O)OCC1)=O c1(C(=O)NCC(C)NC(C2CC(C#N)C2)=O)ccccc1C(=O)N(C)C C1(C(=O)NC2(C)CCN(c3nc(Cl)c(C#N)s3)C2)CC2CCCCN2C1 C1(NC(N2CCN(Cc3ccccc3)CC2)=O)CCCN(C2CC2)C1=O Cc1nc(CNC(=O)Cc2ccccc2F)oc1C(=O)NC1CSCC1C C(CCC(C)(C)C(=O)N1CC=CC(C(N2CCCC(CO)C2)=O)C1)OC c1(C(=O)NC(CC)CNC(=O)CC2CCCCO2)cc(O)n(CC)n1 C12(NC(c3ccn(C(C)C)n3)=O)CCCN(C(=O)C=CC3CCOC3)CC1C2 c1(-c2ccc(C(C)O)s2)c(CN2CCN(CCN3CCCC3)CC2)cnn1C N1(C(Cc2c(C)noc2C)=O)CC2CCN(CCOc3ccccc3C#N)C2C1 N1(C(C(C)c2ccco2)=O)CCCN(C(c2cccc(C(F)F)c2F)=O)C(C)C1 CCCC(C)(C)CC(=O)NCCCN(C)C(c1sccc1C(C)=O)=O c1(CC)c(C(=O)NCC2CN(C(=O)CC(C)F)C(C)(C)C2)sc2ccccc12 C1(CC(=O)N(C2CCCC2)CC=C)CN(C(C2CC(O)C2)=O)CCC1C C12(C(=O)NCc3cnc(C)o3)C(NC(=O)CCC3CC3(F)F)C3CC1C2C3 CCC(CC(=O)NCC(CC(=O)NCC1(O)CCN(C)C1)C1CCC1)C(C)(C)C C1(Oc2ncc(C(=O)Nc3cn(C)nc3C(=O)NC3CC3)nc2)CCCCC1(F)F N1(C(C(C(C)C)(C)C)=O)CCC2(CCCC2NC(C2CN(S(N)(=O)=O)C2)=O)C1 N1(C(COCCCOC)=O)CC2C3CCC(C(NC(c4cscc4Cl)=O)C3)C2C1 C=CCC(C)(C)C(=O)N1CCC(C(C)C(=O)NCC(C)(CC)C(N)=O)CC1 c1(OC)ccc2sc(CN3CCCC3C(C)C(=O)OC)c(C)c2c1 C(CCC)(C(O)C(=O)N1CCCC1CN=[N+]=[N-])NC(C(C=C)O)=O Cc1nc2nccc(NC3CC(C)N(C(=O)C(C)(F)F)C3)n2n1 c1(-c2nc(-c3cc(C)c(C4CC4)cc3)on2)ccc2occ(C)c2c1 N1(C(Cc2c(C)cccc2)=O)CCN(C(c2cc(CO)[nH]n2)=O)C(C)C1C N1(C(C(C)=C(CC)C)=O)CCC2CCC(NC(c3ccccc3OCC)=O)C1C2 C1(NC(c2c(C)n(C)nn2)=O)CCN(C(c2ccnnc2)=O)CC1F N1(C(Cc2cc(C)cc(C)c2)=O)CC(NC(c2coc(Cl)n2)=O)CC12CCC2 c1(C(N2CCC(NC(CC3CCCC(C)O3)=O)(CF)C2)=O)cc(F)cc(F)c1N C1(NC(C2(C)CC2)=O)CC2(C1)CN(C(C1CCCN1C(c1ccccc1)=O)=O)C2 C1(CC(=O)OC)CN(CC23CC(C#N)(CO2)C3)CC2(CCC2)O1 CC1(C(N2CC(NC(=O)CCc3ccc(Cl)cc3)C(O)C2)=O)COCC1(F)F Cc1c(O)ccc(C(N2CCN(C(C34CC(C)(CO3)C4)=O)CC2)=O)c1C C1(F)(C(=O)NCc2cccc(CC)c2)CCCN(C(C2(CO)CCCO2)=O)C1 C(CCCC(C)NC(=O)Cn1nnc(C)n1)NC(C1(COC)CCOC1)=O c1(C(N2CC3(C(NC(CC(CCC)C)=O)CC3)C2)=O)cn(C)c2ccccc12 C1(CNC(C(C)(C)OCCC)=O)CN(C(C2CCOC2CC)=O)CCN1C C(=O)(C(C)(C)C#N)NC(C1CCCN(C(=O)CCSc2ccccc2F)C1)C C1(O)(CNC(c2c(C)nc[nH]2)=O)CCN(C(=O)CC2OCCC2(C)C)C1 c1(C(N2CCOCC(NC(C=COCC)=O)C2)=O)cnc(O)c([N+](=O)[O-])c1 N1(C(COCC(=O)NC)=O)CC2CC(C(=O)NC(CO)CC(F)(F)F)(C2)C1 N1(C(CCCCOCC)=O)CCN(C(=O)C(C)N2CC(C)C2)CC12CCC2 CCCCCC(O)C(=O)N1CCC(NC(c2oc(CCC)nc2C)=O)C1 C1(NC(C2CC(NC(CCCC=C)=O)C(O)C2)=O)CCCC(O)CC1 c1(C(=O)NCC2N(C(C(C)SCC)=O)CC2)cccc(F)n1 c1(C(N(C)CC2N(C(C(C)OCCC=C)=O)CC(F)C2)=O)cccc(N)c1Br N1(C(C2CC(=C)C2)=O)CC2CS(=O)(=O)CC2(CNC(C2(COC)CCC2)=O)C1 N1(C(COC(C)C)=O)CC2(CC(CNC(C3CC4(C3)OCCO4)=O)C2)C1 C(c1cccc(O)c1)=CC(=O)NC1(CN(C(=O)C(C)(C)CO)C)CC1 C1(O)(C(N2CC(NC(c3occc3F)=O)C2)=O)Cc2ccccc2C1 N1(C(CC(OCC)OCC)=O)C2CCC(C(=O)NC(CC)CCO)C1CC2 CCS(=O)(=O)C=CC(=O)N1CC(F)(F)CC1CNC(=O)C(F)Cc1ccccc1 N1(C(c2n(C=C)ncc2)=O)CCN(C(c2coc(S(=O)(=O)NC)c2)=O)CC(O)C1 C1(C(=O)NC(CN(C(C(C)OCCOCC)=O)C)C)CCC(=C(F)F)CC1 Cc1ccc(OCCC(=O)NCC2CCN(C(=O)C=CC3CC3)CC2)cc1C c1(C(=O)NCC2(NC(c3ccc(C(F)F)cc3F)=O)CC2)ccc(O)c(F)c1 c1(C(N2CCCN(C(C(C(=O)OCC)F)=O)CC2)=O)cc2ccc(C)cn2n1 c1(C(=O)NCC2(CNC(CNC(CC)=O)=O)CCC2)ccc(C(=O)NC)c(F)c1 N(C(=NCCF)N1CCCC2(CC2)C1)CC1CN(C(=O)OCc2ccccc2)C1 c1(NC(c2cc(C3(C)CC3)n[nH]2)=O)nn(C)c(Cl)c1Cl.C12(CC1)CN(C)C2 CC1(C(=O)NCC(CO)NC(c2csc(C(F)F)c2)=O)CC(C2CC2)=NO1 C(=O)(C1c2ccccc2OCC1(C)C)N1C(CNC(c2ncc(C)c(Cl)c2)=O)CC1 N1(C(c2ccc(OCC(C)C)cc2)=O)CCN(C(=O)C(O)C(F)F)CC(C)(C)C1 C1(OCC#C)CCCN(C(=O)C(n2cc(-c3cc(C(=O)OC)cs3)nn2)C)C1 CC1CCCC(N(C(=O)NC2CCCCC2)Cc2ccnc(N(C)C)c2)C1 C1(NC(c2c(CC)c[nH]n2)=O)CCCC(N(C)C(C2CC(O)C2)=O)C1 c1(C(C(=O)N(CC(C)NC(=O)C(C)(C)C2CCOCC2)C)C)cccc(C#N)c1 c1(C(N2CCC(C)(N3CCCC3)C2)C(=O)NCC=C)n[nH]c2ccccc12 N1(CC)CCC2(CC1)CC(C(N1CCC(c3nc4ccc(C)cc4[nH]3)CC1)=O)C2 N1(C(C2(OCC)CCCC2)=O)CCC2(CCC(NC(C3(C)CC(F)C3)=O)C2)C1 CN1CCN(CCC(=O)N(CCCNC(C2CCC(O)C2)=O)C)CC1 CS(=O)(=O)C(CN=c1[nH]c(N2CC3CCC3C2)nc2c1SCC2)C1CC1 C1(CNC(=O)C(c2ccccc2)F)CNCCOC1 CON1CCC(C(=O)N(C2CN(C(c3cn(CC(F)F)cn3)=O)CC2F)C)CC1 N1(C(CSCC(=O)OCCCC)=O)CCCC(OC)C1.C1(=O)C(C)NC(=O)N1 C1(C2CC2)(NC(C=CCN(C(C(CC(C)C)=O)=O)C)=O)CCCCC1 CC1CC(NC(=O)CN2CCS(=O)(=O)CC2)CCN1C(c1nncs1)=O c1(C(=O)NCCCN(C(C(=O)NCC)=O)C2CCCC2)c(C)nc2sccn12 c1(NCCc2c(C)cccn2)cc(Br)ccc1S(=O)(=O)N1CCN(C=O)CC1 N1(C(CCCCCOCC)=O)CCC2(CNC(c3ncccc3Cl)=O)CCCC12 c1(COC)nc(NCC2(OC(C)C)CCOC2)cc(=NCc2ccc(Cl)nc2C)[nH]1 CCCC(CC)C(=O)NC(CCSC)C(=O)NCCN1CCCC1 c1(C(=O)NC2CCCN(C(C=CCC)=O)CC2)ccccc1S(C)(=O)=O C1(CCNC(c2ccccn2)=O)CSCCN1C(=O)CNC(=O)C(F)(F)F c1(CC)ccc(N)c(C(=O)NC2CCCC2NC(=O)C=CC2CCOCC2)c1 C1(C(N(CCCCCNC(C2(SC)CCC2)=O)C)=O)CC2C=CCC(C1)C2 C1(C(N2CCC(C(C)NC(=O)C(F)C3CCOC3)C2)=O)(CC)CCOCC1 C1(Cc2n(-c3cc(F)cc(F)c3)nc(COC(F)F)n2)CCn2nccc2C1 N1(C(C2N(C(=O)OC(C)(C)C)C(C3CC3)CC2)=O)CC2COCC2(CO)C1 c1(OC)nccc(C(=O)NC2CC(CC(=O)NCC(C)O)C2)n1 c1(C(=O)NCCCC(C)NC(CCSC)=O)cnc(Br)c(N)c1 CC1=CCC(C)(C(N2CC3C(NC(c4cnn(C5CC5)c4)=O)C3C2)=O)CC1 C1(N(C)C(c2cc(-c3ccc(F)cc3)[nH]n2)=O)CC2CC1N(C(=O)C(N)=O)C2 c1(C(N2CC(CC(C)NC(CNS(NC)(=O)=O)=O)C2)=O)ncc(N)cc1Cl N1(C(CC2CC(OC)C2)=O)CCC(NC(c2cnc(S)[nH]2)=O)C(F)(F)CC1 CCCCC(C(=O)NC(C)CC1CN(c2cc(C(=O)OC)nc(C)n2)C1)C(C)C CCC(C)CCCCC(=O)N1CCOCCC1C(=O)NCCCc1ccccn1 N1(C(c2onc(C)n2)=O)CCCCC(C2CN(C(=O)CCC3CC(F)(F)C3)C2)C1 C#Cc1cccc(CC(=O)N(C)CC2CCCN(C(=O)C(=O)C(C)(C)C)C2)c1 c1(C(N2CC3CC(NC(C4CC=CC4)=O)CC3C2)=O)cnnc2ccccc12 N1(C(CCCN(C(=O)CCC(=O)C2CC2)C)=O)CCCNC(=O)C1 N1(C(c2cc(C)c(C)s2)=O)C2CC=C(C(=O)N3CCC(F)(CF)C3)C1CC2 C(c1cncc(O)c1)=CC(=O)NCCCOCCNC(C1CSCCS1)=O c1(C(=O)NCC23CC(NC(C=C4CCC(C)CC4)=O)(C2)C3)cnc2c(c1)CCC2 N1(C(CCN(CCC)C)=O)C2CCC1CC(C(=O)NCc1ccnc(OC)c1)C2 c1(C(C(=O)Nc2ccc(F)cc2)N(C(CC)COC)C)cnn(C)c1Cl C1(NC(C(CC)n2ccnc2)=O)C(C)CCN(C(c2cnc(O)n2C)=O)C1C Cc1c(C(N2CCOC(C(C)NC(=O)C3=CC(C)(C)C3)C2)=O)cncc1Br C1(N(C(C(CC)O)=O)CC(C)C)CCN(C(C2CN(C(C)=O)C2)=O)CC1 C1(NC(c2ccc3c(c2)CC3)=O)CN(C(=O)COCC2CCOC2)CCC1F c1(OC)ccsc1C(=O)NCc1cccnc1.C1(C)C=CC(=O)N1C1CC1 C1(C)(C(=O)NCC2(F)CCN(C(C(C(C)C)N(C)C)=O)C2)CC(C(C)C)=NO1 C#Cc1cccc(C(=O)NCC(O)CNC(c2cnccc2C(C)(C)C)=O)c1 N1(C(C(C)(C)Oc2ccccc2)=O)CCCCC1CNC(c1ccoc1Cl)=O C1(C(N2CC(O)(CNC(=O)CCOc3ccc(F)cc3)C2)=O)CC2C=CC1CC2 CCCCCC(O)CC(=O)NC1CCCC(NC(=O)CCCCn2ccnn2)C1 c1(OC)ncnc(OC)c1C(=O)NCC(C)(C)CNC(=O)C=Cc1cn(C)nn1 c1(C(=O)NC2C(C(N3CCC(CC)(CO)CC3)=O)OCC2)ccc2occc2c1 c1(C(c2n(CC(=C)C)nnn2)NC2(C(=O)N(C)C)CC2)nc(C)sc1C c1(CNCCc2nnn(C(F)(F)F)n2)ccc(I)cc1 C(=O)(C1CCCc2nncn21)NC1(CO)CCCN(C(CCSCC(C)C)=O)C1 Cc1nc(C(=O)NCC2(NC(=O)CSc3nccn3C)CCC2)c2ccnc-2[nH]1 c1(NC(C(Cc2cc[nH]n2)NC(c2cc(Cl)cs2)=O)=O)ccccc1Cl N1(C(Cc2c(C)nc(O)nc2C)=O)CC2CCC(C1)N(C(=O)CC(C)(F)F)C2 c1(C(=O)NC(CC)CN(C(=O)CC2COCCO2)CC)sc2cccnc2c1Cl C(CC(C(C)(C)C)NC(c1ncnc(O)c1Cl)=O)N(C(C(CC)(C)O)=O)C N1(C(C(CC)Oc2ccccc2)=O)CC2CC2(NC(c2[nH]nnc2COC)=O)C1 c1(NCC2(OC)CCCS(=O)(=O)C2)ccn2ncc(S(C)(=O)=O)c2n1 N1(C(C2(OC)CCC2)=O)CCC(O)(CCNC(C2CC2C(C)C)=O)C1 C(C(C)C(C)C(=O)NC1(CNC(C2CCCN(C)C2)=O)CC1)OC N1(C(Cc2c(C)nccc2)=O)CCC(C)C(NC(=O)CCC2CCCCC2)C1 C1(C(N(CC(C)(C)NC(c2c[nH]nc2C2CC2)=O)C)=O)CCCCC(F)(F)C1 C1(CC(=O)N(C)CC2N(C(COCC(=O)NC)=O)CCC2)CCOC1(C)C N1(C(COC)=O)CCCC(C)(C(=O)Nc2cnncc2Br)C1 N1(C(c2nc(NC(C)=O)sc2)=O)CCOCC(F)(CNC(C2(CO)CC2)=O)C1 C(CNC(=O)CP(C)(C)=O)(CC(F)(F)F)NC(Cc1nnc(C)o1)=O CCCCC(C)(F)C(=O)NC1CC2CC(C1)N(C(=O)Cn1cnc([N+](=O)[O-])n1)C2 N1(C(c2c(CCCC)ocn2)=O)CC2(CC(NC(=O)C(C)CN(CC)CC)C2)C1 C1(C(=O)NCC2(O)CCC(C)C2)(NC(C2CCO2)=O)CCc2cc(Br)ccc2C1 C(C)(CNC(C1CC(C(F)(F)F)(OC)C1)=O)(C(C)C)NC(C=C(COC)C)=O C1(C)(C(=O)OCC)CCC(C(F)(F)F)CC1.C1(C)C(=O)N1C1CC1 CC1=C(C(=O)N2CCCC(N(C(=O)CC3NC(=O)NC3=O)C)CC2)CCO1 c1(C(=O)OC)cc(C)cnc1NC(=O)C(=O)NCCN(CCNCCO)C c1(OC)cc(C(=O)NC2CC(CC(=O)NCC(N)=O)C2)ncn1 c1(OC)ccc(C(=O)NC2CCC(N(C(=O)CSCC3(F)CC3)C)C2)nn1 N1(C(c2ccc(-c3n(C)ncn3)cc2)=O)CCCC(NC(=O)CC(F)(F)F)C(F)C1 c1(C(=O)NCCNC(C2(C)CCSCC2)=O)ccn2ccnc2c1 C(CCCCC(=O)N1CC(COC)CC1CNC(c1cccc(Cl)c1)=O)=CC C1(C(=O)NC(C(=O)N(CC(C)C(C)(C)C)C)CCC2CC2)CC2(CCC2O)C1 Nc1cc(-c2cn(CCC3CC(NC(c4sccc4CO)=O)C3)nn2)ccc1Cl c1(C(=O)NCCCNC(c2c(C)n(CCO)cc2)=O)nc(Cl)c(Cl)c(N)c1Cl c1(NC(CC)CO)cccc(NC(C2CCC2)=O)n1 CC1CCCn2c(C(N3CCN(C(C4CCC(C)(C)C4)=O)CC3C)=O)cnc21 C1(C(N2C(C)(C)C(CNC(=O)CC3CCCC3)CC2)=O)COC2(CCC2)CO1 c1(CC)[nH]c(=N)sc1C(=O)NC1CCC(N(C)C(C2CC=CC2)=O)C1 C(c1ccco1)=C(C)C(N1CCC(N(C)C(c2cnnn2C)=O)C1)=O c1(NC(C(CCO)OC(c2c(C(=O)OCC)scc2)=O)=O)ccc2c(c1)OCO2 Cc1nc(CO)sc1C(=O)NC1CCOCC1NC(C1CC(O)C1)=O CC1CN(C(=O)C(=O)NC2CC2)CC1NC(c1ccc(CN2CCCC2)cc1)=O c1(C(N2CC(CC(C)NC(c3ncccc3F)=O)C2)=O)cc([N+](=O)[O-])nn1C N1(C(c2ccc(C)n2C)=O)CC2OCC(NC(C3CCN(C)CC3)=O)C2C1 N1(C(c2c(C)nccn2)=O)CCC(CNC(=O)C(C)O)CC1C C(=O)(CCS(N)(=O)=O)NC(C(C)C)CCNC(=O)Cc1cc(C(F)(F)F)n[nH]1 c1(C(N2CC(O)(CCNC(C3CCCC(C)O3)=O)C2)=O)ccc2[nH]ccc2c1 CCCCCC(O)CC(=O)NC(C)CN(C)C(C1CCOC(CCC)C1)=O N1(C(C(n2c(C)ncc2)C)=O)CC2(CNC(C3CCCC(F)C3)=O)CC(F)(C1)C2 C1(OCc2c(C(=O)OC)[nH]nc2Cl)CCc2cc(OC)ccc2C1=O c1(C(=O)NC(C2OCCN(C(CCC(=O)NC)=O)C2)C)ccc([N+](=O)[O-])n1C c1(OC)ccc2c(C(=O)NC3CCN(C(=O)C#CC4CC4)CC3F)csc2c1 c1(C(=O)NC(CC2CN(C(C(CC#C)O)=O)C2)C)ccc2ccn(C)c2c1 N1(CCC(CCC)C)CCCSC1=Nc1ccncc1OC c1(OC)cc(C(=O)NC(CCN(C(=O)C(O)C2CCCC2)C)C(C)C)cc(C)n1 C(CS(=O)(=O)c1ccc(C)cc1)NC(c1cc(F)ccc1F)CC=C c1(OC)cc(C(N2CCC3(NC(=O)C4=CCCC4)CCCC23)=O)cc2c1OCC2 C(=O)(C1=CC2C=CC(C1)C2)NC12CC(NC(c3cnc4ccsc4c3)=O)(C1)C2 c1(CC(=O)NCCN(C(=O)C=CCOCC)CCC)nc2ncccn2n1 CN1C(=O)Cc2ccc(C(=O)NCC3(C)CCN(C(C4COC(=O)N4)=O)C3)cc21 N1(Cc2cccc(CC)c2)CC(NC(c2ccc(OC)nc2OC)=O)C(C#N)C1 c1(C(N(C(C)C)CCNC(c2ccn(C)c2)=O)=O)ccc(Cl)c(Cl)c1N c1(CNC2CCC(NC(C3(C(F)(F)F)CCC3)=O)C2)cc(Br)ccc1OC(F)(F)F Cc1ccc(C(C(=O)NC(C(=O)O)c2cccs2)C2CC2)cc1 N1(C(c2c(CCC)n(-c3ccccn3)nc2)=O)CCCC2CC3(CCC3)C12 c1(C(=O)NCCC2N(C(CCC#C)=O)CCOC2)cnc2c(C)cnn2c1 c1(C(=O)NCCCN(C)C(c2cccc(N)c2F)=O)cc2cc(F)ccc2s1 c1(CC(=O)NC2CC(C(=O)Nc3nnc(C(C)(C)C)s3)C2)ccc(Cl)cc1 C(CC1CCC1)(C(=O)NCC(F)CO)NC(CSCCCC)=O Cc1conc1C(=O)NC(C(=O)NC1CC1F)c1ccoc1 Cc1ccc(NC(=O)C(CC(C)C)ONC(C2CCC(C3CC3)C2)=O)cc1F c1(CC)n[nH]c(=NCC2(NC(=O)Cc3cccc(COC)c3)CCC2)o1 C=CC(CCC)CC(=O)N1CCCC1CN(C(=O)COc1cc(F)cc(F)c1)CC Cc1n[nH]cc1NC(c1nc(C(=O)NCc2ccoc2)cs1)=O C1(CCNC(c2n(CC)ncc2)=O)CC(OC)CN1C(c1cocn1)=O Cc1c(C(=O)NCC(C)CNC(c2cnc(C3CCOC3)s2)=O)cccc1C#N N1(C(CCN(CC=C)C(C2CC2(Cl)Cl)=O)=O)CC(F)CC(F)C1 N1(C(CCC(=O)NCC)=O)CCCC2CCN(C(C3CS(=O)(=O)C3)=O)CC12 C(=O)(C(CC1CC1)Nc1ccc(C(F)F)s1)NCC(OC)OC N1(C(C2C(=C)C2)=O)CCCC2(CCN(C(c3ncoc3CC)=O)C2)C1 CC(CCNC(c1cnc[nH]c1=N)=O)CCNC(c1ccc(C2CCC2)nc1)=O CC(C)=C=CC(=O)NC(Cc1cc[nH]n1)C(=O)NCC1CCC=CCC1 c1(C(N2C(CNC(CC3C(OC)CC3)=O)CC2)=O)nc(C)ns1 CCC(CC)CCCN(C)C(C1CC(C)N1C(=O)C=Cc1cc(C)no1)=O c1(NC(C2(C)CCCN(C(Cc3c(C)cccc3)=O)C2)=O)nc(Cl)c(Cl)cc1Cl C1(C(N2CC(C)(CC)C2)=O)CC2CC1CN(C(C1(CO)CC1)=O)C2 C1(NCC2CC(NC(COCCCOC)=O)C2)CC2(CC2)C1.C1C(=O)N1 C12(c3cn(C(c4ccccn4)C)nn3)CC(CN1C(=O)NC1(C)CCOCC1)C2 C(N=c1nc2ncn(C)c2c(NCc2cc(C(F)F)no2)[nH]1)c1nnn(C)n1 N(C(=NCCCSC)NC1CCN(c2nccs2)CC1)CC1(OC)CCSCC1 c1(C(=O)NCC(C)CN(C)C(C2(C)CCC(=O)C2)=O)ccnnc1O C1(N(C(=O)CCSCC(N)=O)C)CCCCN(C(=O)C=CC(=O)N(C)C)C1 C=C1CC(C)(NC(c2nnnn2CC2CC2)C2CC3(CC3)C2)C1 Cc1cccc2c(C(=O)NC3CCCC(NC(C4CC4C)=O)C3)cccc12 N1(C(c2cncc(NC)c2)=O)CCC(CNC(c2c(C)noc2C)=O)C12CC2 c1(C(N2C3CN(C(C(=O)N(C)C)=O)C(CC3)C2)=O)cc2cc(Br)cnc2[nH]1 c1(N(C(c2cnn(C)c2)C(=O)NC(CC)(C)C)C)ccc(N(C)C)cc1OC CC(C)(C(=O)NCC1CCCN1C(=O)CC1CC=CCC1)N1CCOCC1 N1(C(C2CCN(C)CC2)=O)CC(NC(C2CCS2(=O)=O)=O)C(C2CC2)C1 c1(CC(=O)NCC2C(NC(c3n(C)nnc3Br)=O)C2)ccc2occc2c1 C1(C)(C(C)NC(C2CCCO2)=O)CN(C(=O)C(C)Sc2nncn2C)C1 N1(C(CC2N(C(C(C)(C3(C)CC3)OC)=O)CCOC2)=O)C2C=CCC1CCC2 C1(NC(C2(C(F)(F)F)CCC2)=O)CCCC(NC(C2(C(F)F)CCCO2)=O)C1 c1(C(=O)NCC(CNC(Cn2c(C)nnn2)=O)CO)ncccc1N(C)C C1(CNC(C=CC(C)C)=O)CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CCC1C c1(CC)ccc2occ(C(N3CC(NC(=O)C(O)CC)C(C)(C)C3)=O)c2c1 CC1(C)CN(C(c2ccn(C(F)(F)F)n2)=O)CCC1NC(=O)Cc1ccno1 C12(C(=O)NC(C)(C)CNC(C3CC34CCC4)=O)CCCCC1NC(=O)CC2 c1(CN2CCC(=O)N(CC(CC(F)(F)F)N3CCC3)C2=O)nc2cccc(Cl)c2[nH]1 c1(C(C)=O)ccc(NC(=O)CC2CCCCN2C(N2CCCC2)=O)cc1C c1(OC)ccc(C)c(CNC(=O)NC2CCOC(C(C)C)C2)n1 CC(C)C(O)CC(=O)N1CC=CC1(C)C(=O)NC(c1nn[nH]n1)C1CC1 c1(C(N2CCC(NC(CCCC=C)=O)C(F)C2)=O)ccc2[nH]c(=N)sc2c1 CCC(O)C(C)(C)C(=O)NOCC(=O)N(C)CC1(C)CCCO1 C1(CN(C(CSCCC)=O)C)CC(F)CN1C(=O)Cn1nnnc1-c1ccsc1 C1(CC)CN(C(=O)C(F)(F)c2ccnn2C)CCC1NC(c1cccc(O)n1)=O c1(CO)cccc(CN=c2[nH]nc(Cl)s2)c1F CCCCCC(C(=O)NCC1CCCN(C(=O)C(C#N)CC)C1)C(C)C N1(C(C=Cc2ncc(C)[nH]2)=O)CCC(C)(NC(c2cc(O)ccc2Br)=O)CC1 C1(NC(c2n[nH]cc2F)=O)CCN(C(=O)C=CC2CCOC2)CC1F O=C1NC(=O)c2ccccc2C1=CNC(c1ccc(C2CCCC2)cc1)=O c1(C(C)O)ccccc1NC(=O)C=CCN(C)C(c1ccsn1)=O CC1(C)COCCC1C(=O)NCC1CCN1C(c1ccc(C(N)=O)[nH]1)=O C1(C(=O)NCCC2(OC)CN(C(=O)C=Cc3nnn(C)n3)C2)CC1C1CC1C Cc1ccc(C(C)NC(c2ccc(F)cc2)c2nnnn2C2CCOCC2)nc1 C(=O)(C(CN(C)C)C(C)C)N(CC(CC)NC(c1nc(Cl)ccc1N)=O)C C1(NC(C2C(C)C2)=O)CCCCN(C(=O)CCSc2ccc([N+](=O)[O-])cc2)CC1 N(C(=NCCF)NCC(CO)CC(C)C)C1CCN(CCOC)CC1 c1(C(C(=O)NCC2CC(n3cc(C4CCCC(O)C4)nn3)C2)O)ccc(Cl)c(Cl)c1 c1(C(N2CC3C(CNC(C(C)C4CC4)=O)(CC3)C2)=O)cc2occ(Br)c2[nH]1 C(C)(C(C(C)C)NC(=O)CSCc1cscn1)NC(c1cc(CC)sc1)=O C1(C2(NC(C3CCC3(F)F)=O)CC2)CCCN1C(c1ccsc1Br)=O C1(C2CCCCO2)(C(=O)NCCNC(=O)C(c2ccccc2F)O)CCOCC1 C1(NC(c2c(CC)n(C)nn2)=O)CCN(C(c2cc(C)nn2C)=O)CC1C CC1CC(CNC(C2CCN(CC(F)F)CC2)=O)CN1C(=O)C=CC1CCOC1 c1(C(N2CCC(F)(C(=O)Nc3c(C)cnc(Cl)c3)C2)=O)cc(Br)c2cc[nH]c2c1 C1(NC(C)(C)C)COC2CN(C(=O)O)CC12.c1(CNC(C)=O)c(Br)noc1C1CC1 C1(CNC(C2C(CCC)CCC2)=O)CN(C(=O)CNc2ccccc2)CCCO1 N1(C(c2c(OC)nccc2)=O)CC(CC(=O)NCCCc2nccs2)CC1(C)C N1(C(C2(C(C)C)CCC2)=O)CCCCC(CC(N2CC(O)(c3nn[nH]n3)C2)=O)C1 c1(C(N(CCC)CCNC(C2CC2(C)C(C)C)=O)=O)cnn(C)c1-n1cccc1 c1(C(N(CCNC(C(C)OCCC=C)=O)C)=O)c(C)nn2c1CCCC2C C1(C(=O)NC(CC)CO)CC2CCC1N2C(C1CCN(c2ccccn2)CC1)=O Cc1cc(CN(C(=O)C(CO)NC(C2CC(=C3CC3)C2)=O)C)no1 N1(C(C2C(C(C)C)C2)=O)CC(CNC(=O)CCc2ccsc2)C2(CC2)C1 CC1CCC(NC(=O)C(c2cccc(Cl)c2)O)CN1C(=O)CN1CCCS1(=O)=O N1(C(C2(COC)CCCO2)=O)CCCC(CO)(NC(c2cnc(C(C)C)s2)=O)C1 N1(C(CCC(C)OC)=O)CCN(C(c2c(O)cccc2F)=O)CC(O)C1 O=C1CCC2CN(C(=O)NC(c3cccc(OC(F)F)c3)C(F)(F)F)CC2N1 C1(NC(c2ccn(C)c2CC(=O)O)=O)CN(Cc2cnc(Cl)nc2Cl)CC1(F)F N(C1CCc2cc(Cl)ccc21)C(=O)NC(c1ccc(Br)cc1)CC N(S(=O)(=O)N1CCCCC1)NC(c1nc(CC)c(-c2ccccc2)o1)C N1(C(c2c(C)nc(C)[nH]2)=O)CCC(C2CN(C(=O)C(O)C3CC3)C2)CC1 CC(C)(CCS(C)(=O)=O)C(=O)N1CCCN(C(=O)CC2CCOC2=O)CC1 C1(CC(=O)NCC(CN(C)C(c2ccc(C3CC3)cc2)=O)O)NC(=O)NC1=O O=C(C#CC1CC(F)(F)C1)NCC12CC1CN(C(=O)CCSC1CCCC1)C2 C1(CNC(C(C)=C2CC2)=O)CC2CCC(C1)N2C(C1CCCCCC1)=O N1(C(C=C(CC)C)=O)CCOC2(CCN(C(=O)CCOC3CCCCCC3)C2)C1 C1(NC(=O)CCN2CCC2)CCCN(C(C2CC3CCC(C2)O3)=O)CC1 C(=O)(C(F)CCC(C)C)NCC1CCCN(C(c2cncc(C#C)c2)=O)C1 N1(C(COCCCCC)=O)CCCCC1C(=O)Nc1[nH]ccc1CC C1(C(=O)NCC2C(CNC(c3cc(C(C)(C)C)on3)=O)C2)C2(CC2)C12CC2 C(=O)(C(C(C)C)c1cnn(C)c1)NCC1(NC(c2c(SC)csc2)=O)CCOC1 N1(C(C2N(CC)CCOC2)=O)CC(NC(=O)C(F)(F)C(F)F)CCC(O)C1 Cc1cc(F)cc(C(=O)NC23CCCN(C(=O)C(C)NS(C)(=O)=O)CC2C3)c1N Cc1cc(F)c(C(=O)NCC2(CCNC(C3C4CS(=O)(=O)CC34)=O)CC2)cc1F CCCCS(=O)(=O)NCC(=O)N(CCCCCN(C)C(C1CC1F)=O)C(C)C C1(C(N2C(C3CCCN(C(CSCC=C)=O)C3)CCC2)=O)CC2(C1)CC(F)C2 N1(C(CCC=CC)=O)CCN(C(=O)C(C)NC(C2CCCC2)=O)CCC1C C=C=CCCC(=O)NCCn1cc(C(=O)NCc2nc(C)cs2)cn1 c1(CCNC(C(CC2CC2)NC(C(CC2CCC2)OC)=O)=O)ncccc1F O=C(C1=Cc2ccccc2C1)NCC1(C(N)=O)CN(C(C2C3CC4C(C3)C24)=O)C1 N1(C(c2c(C)n(C)cn2)=O)CC2CC(C1)N(C(=O)Cn1ncccc1=O)C2 CC1CC(C(=O)NCC(=O)NC2CC2)CN1C.C12(CCC1)C(=O)NC2 Cc1cnc2c(C(=O)NC3CCN(C(c4cncn4C4CC4)=O)C3)cnn2c1 C12(NC(c3cccc(C)c3F)=O)CCN(C(c3cccc(O)n3)=O)CCC1C2 N1(CC)CC(C(N2CCCCC2C(=O)N(CCCCCO)C)=O)CC1=O Cc1cc(C2CC2)ncc1C(N1CCOCC1CCNC(c1ncn(C)n1)=O)=O CCC(CC)(CN=c1[nH]cncc1I)NC(=O)C(C)COC C1(NC(CCCCOC)=O)CCN(C(=O)Cc2cccnc2)CC(C)(C)C1 c1(CC(C)C)cccc(C(=O)NCC(O)CNC(=O)C(O)CN2CCOCC2)c1 Cc1cc(N2CCN(c3nc[nH]n3)CC2)nc(=NC(C)CC(C)(C)C)[nH]1 C1(C#N)(OC)CC(C(=O)NCCCCCCn2cc(-c3ccncc3)nn2)C1 C1(C(=O)NC2CC3CC(NC(CCC)=O)CC3C2)CC2CCC1CC2(F)F c1(NCC2(CNC(C(C=C)(C)CC)=O)CCC2)ncnc2cnccc12 c1(C(=O)NCC2CN(C(CNS(CC)(=O)=O)=O)CC2C)cncc(C)c1C c1(C(N(CCCNC(Cc2scc(C)c2)=O)C2CC2)=O)ccc2c(n1)OCCO2 C1(C(N2CC(CCNC(c3cc(CC)no3)=O)C2)=O)CC2CCCC(C1)C2(F)F CCC(O)C(C)(C)C(=O)N(CCNC(=O)C(c1ccccc1)SC)CC C(=O)(C(F)C(C)(C)O)NC(c1ccc(CNC(C2CCNC2=O)=O)cc1)C Cc1cc(F)ccc1C(=O)NCC1CN(C)CCN1C(=O)CCCc1cnn[nH]1 NS(=O)(=O)c1ccc(NCC2(c3ccccc3)CCCC2)cc1 C12(C(=O)OC)CCC(NC(C3CC3CNC(c3cnns3)=O)=O)(CC1)CO2 C1(CCC)(NC(c2n(CC=C)ccn2)=O)CCCN(C(c2ccc(C)s2)=O)C1 C1(CCOC)CN(C(c2cnc(C3CCC3)s2)=O)CCN1C(=O)C(O)C1CCC1 N1(C(C2(C#N)C(C)(C)C2)=O)CCCC(CO)(CNC(=O)CCc2cccnc2)C1 C12(NC(c3cc(CC)c(F)cc3)=O)CCCC1N(C(=O)C1=C(Cl)CCOC1)CC2 CC1(C)CCCC1CCNC(=O)NCCC1(c2ccccc2)CCCO1 N1(C(c2cc(C)[nH]c2)=O)CCCC(C2CN(Cc3ccc(C(C)(C)C)cc3)C2)C1 c1(C(=O)NCC(C#C)OC)[nH]ccc1CNC(=O)C(C)C N1(C(C(CC)C2CCOCC2)=O)CCC(CNC(c2ccncc2)=O)C(F)(F)C1 CCC(C(=O)OC)C(=O)N1CCN(C(C2CCN(c3ccccc3)C2)=O)CC1C c1(C(=O)NC2C(NC(C(=O)NCC)=O)CCCC2)nn(C)c2c1CSCC2 CC(C(=O)NCC1CN(C(=O)C=Cc2ccncn2)C1)C(C)S(C)(=O)=O c1(NC(CC2C=CC(NC(=O)CCC3CCCC3)C2)=O)ccc2ncnn2c1 N1(C(c2c(O)nnc(C)c2C)=O)CCCCC2(C1)CN(C(=O)CC1=CCCC1)C2 c1(OC)ccc(C(=O)NC2(CO)CCN(C(C3CC(OC)C3)=O)C2)nc1Br c1(C(N(CCCNC(CC(CC)C)=O)C)=O)cccc(C)c1N N1(C(Cc2cccc(SC)c2)=O)CCC12CCN(Cc1cc[nH]n1)CC2 C1(O)(C(C)NC(c2nnc(C)s2)=O)CCN(C(=O)CCCc2cccs2)C1 C1(C)(CCNC(CCC2(C)CC2)=O)CCN(C(=O)Cc2ccco2)CC1 c1(CC(=O)NC(CNC(C2CC(O)(CC#C)C2)=O)CO)ccccc1SC N1(C(CC(CN(C)C)O)=O)CCC(C)(C)C(CNC(=O)CCSCC(N)=O)C1 N1(C(c2ccc(C(F)F)cn2)=O)CCN(C(=O)CO)C(c2ccccc2Cl)C1 C(=O)(C(C)(C)CCC#N)NCC(Cn1cc(CNC(C(C)O)=O)nn1)(C)C C1(C(=O)OC(C)(C)C)CCOC2(CCSCC2)C1.C1(OC)CN2CC1NC(=O)C2=O Cc1cnc(C(N2CC(CNC(c3cccc(C(F)F)c3)=O)C2)=O)c(F)c1 Cc1ccncc1CCNC(C1CC(NC(=O)CCCCC2CC2)C1(C)C)=O C1(NC(CC(C)C)=O)CCN(C(=O)C(C(C)C)n2ccnc2)CC1 CC1(C)COC(C(N2CC(O)(CCNC(=O)CC3CCC(C)CC3)C2)=O)C1 n1(C(CC)C)nccc1C(=O)NC(c1cn(CC2CCC2(F)F)nn1)(C)C Cc1[nH]nc2c(C(=O)NC3CC3CNC(c3ncccc3C3CC3)=O)cccc12 Cc1nc(C(C)C)ncc1C(=O)NC(CNC(=O)CN1CC(C)C1)C(C)C(C)C CCC(CC(F)(F)F)C(=O)N(C)CCOCCCNC(=O)C(C(=O)OC)C1CC1 C1(=CC(=O)NCC=CCNC(CC2C(C)CCO2)=O)CCCCC1(C)C C1(CC(=O)NCc2cccc(C#C)c2)CCC(C)(C)N(C(=O)C=CCCC(C)C)C1 c1(CC)ncc(C(N2CC(c3ccc(C)cc3)CC2C)C(=O)NC2CCC2)cn1 c1(COC)ccnc(C(=O)NCC2(F)CN(C(c3coc(C)c3)=O)C2)c1 C1(C(N2CC(C3OCCN(C(C4C(CC)CCC4)=O)C3)C2)=O)CC(C)(C)CCO1 c1(C(N2C(C(C)C)(C(=O)NCCC3(C)CC3(F)F)CCC2)=O)cc(O)nc(O)n1 Cc1ncccc1CC(=O)N(CCC(=O)NCC1CC1C)C c1(C(N2CCCC(CNC(C(CCC)NC(N)=O)=O)C2)=O)ncc2ccccn12 c1(C(=O)NC2CC(C)N(C(c3ccc(Cl)[nH]3)=O)CC2)cncc2ccccc12 N1(C(CC(=O)NCC)=O)CCC(CNC(C2(Cl)CC2)=O)C(C)C1 c1(CNC(c2cc3ccccn3c2)=O)nc2c(s1)CN(C(c1cscn1)=O)CC2 c1(C(=O)NCC2C(NC(C(C)NC(C)=O)=O)CC2)ccc(O)c(Cl)n1 C(C1=NOC2CN(C(=O)CCCS(N)(=O)=O)CC12)NC(c1noc(CC)c1C)=O C1(C(=O)NCC2C(C)CN(C(=O)CC3(O)CCOCC3)C2)CC2(CCCC2)CO1 C1(C(N(CC#C)Cc2ccco2)=O)CCC(C(C)C)N1C(C1CCCC(=O)N1)=O N1(C(C(CC)CC)=O)CCN(C(C2(C#N)CCCCC2)=O)C2(CC2)C1 c1(C(=O)NC2CN(C(CSCC(C)C)=O)CC(C)C2)cc(C#N)c(O)nc1N c1(OC)ccc(Cl)c(F)c1-c1cn(CC(=O)OC2(c3ccncc3F)CCC2)nn1 n1(CC(N2CC(CC(C)NC(C3C(C=C)C3)=O)C2)=O)c(=O)oc2ccccc12 C#Cc1cnc(C(=O)NCCN(C(=O)C(C(C)C)C(C)C)CC)c(C)c1 N1(C(C2CCC(C)C2)=O)CCCCC2(CCN(C(c3ccc(Br)o3)=O)C2)C1 C1(NC(CCSCC)=O)CN(C(=O)Cc2cnns2)C(C)(COC)C1 C(=O)(C1=NOC(C2(O)COC2)C1)NC(CNC(c1cc(C)ncc1)=O)C1CC1 N1(C(c2nc(CC)oc2)=O)CC2CC1C2CNC(=O)CC1(O)CCC1 Cc1cc(C)c(C(N2CC(CCCCNC(c3nccnc3N)=O)C2)=O)s1 CC1(C)C(NC(=O)CNC(=O)Cc2ccno2)C(C)(C)C1C(N1CCOCC1)=O c1(CCNC(C(C2(C)CC2)NC(C2C(CC)OCC2)=O)=O)cnn(C)c1C C1(C)(CC)CC(C(=O)NCCC=Cc2ccc(OC(F)(F)F)cc2)CCO1 N1(C(C=C(C)C(C)C)=O)CCCN(C(=O)CCOc2cccc(C)c2)CC1 c1(C(=O)NCC2(O)CN(C(=O)C=C3CCCC3)C2)csc(Br)c1Cl CCC(O)C(C)(C)C(=O)NC1CCC1CNC(=O)CCc1ccnn1C Cc1cc(C(=O)NC2CN(C(=O)C=CS(C)=O)C2)c(F)cc1F C1(C(=O)NCC2(NC(=O)Cc3nc([N+](=O)[O-])n[nH]3)CCC2)CCN2CCOCC12 C(=O)(C(F)(F)C(F)(F)F)NCC(CNC(c1cccc(N2CC=CC2)c1)=O)O c1(C(N2C3C(NC(CCCOCCC)=O)CC(C3)C2)=O)ccc2oc(=N)[nH]c2c1 c1(N2CCn3c(O)nnc3C2)nc(N2CCCC(F)C2)nc2ccc(Cl)cc12 c1(CC)onc(C)c1C(=O)NC(C)CC(C)NC(C1(CC)CC(C)(C)C1)=O C1(C(N(CCCNC(c2nc(C)sc2)=O)Cc2ccccc2)=O)CNC(=O)N1C C(C(C(C)C(C)C)NC(c1cnc(C(C)(C)C)[nH]1)=O)NC(C1CC(=C)C1)=O C1(C(=O)NCC(CC)(CC)NC(c2c(CC)c[nH]c2)=O)CCc2c(n[nH]c2C)C1 C1(C(C)(C)C)CCN(C(=O)C2=NOCC2)C(CNC(C2(C3CCC3)CC2)=O)C1 C=CCCCCCCCC(=O)N(CC(C)NC(c1cn2cc(C)ccc2n1)=O)C N1(C(C2(C#N)CC3(CC3)C2)=O)Cc2nccn2CC(NC(C2CC23CCC3)=O)C1 C(=O)(C(C)(F)C(=O)N(C)CCC1CCN(C(C2CN(C(C)=O)C2)=O)CC1)OC C(C)(CO)(C(=O)N1CCCC(C(C)NC(=O)CCCOC(C)C)C1)OC n1(C(C)C)nc(Br)cc1C(c1nnnn1C)NCc1cccc(O)c1 Cc1ccc(C(=O)NCC(C(=O)NC2CC23CCOCC3)C(C)C)c(C)c1 c1(C(=O)NC2C=CCN(C(Cc3ccc(C)s3)=O)C2)ccc2ccnc(O)c2n1 C(C(C)(C(=O)NC(C)CCN(C(=O)C(O)C1CC1)C)OC(=O)NC(C)(C)C)SC C1(CC(N)=O)(NC(C(C)OCC#C)=O)CCN(C(C2CCCC(C)(C)C2)=O)CC1 Cc1cc2[nH]c(C(=O)OC(C(F)(F)F)C3CC3)cc2o1 Cc1cccc(C)c1OCC(=O)NC1CCN(Cc2cc(CC3CC3)on2)CC1C c1(OC)cccc(Br)c1C(N1CC2(CC(C(N3CCC(C)C3)=O)C2)C1)=O c1(NC(CCNC(c2c(C)c[nH]n2)=O)=O)cccc2ccncc12 c1(C(=O)NCC2C(CNC(c3cncs3)=O)C2)c[nH]c2ccc(Cl)cc2c1=O Cc1cc(NC(C2CN(Cc3ccccc3C(=O)O)CCO2)=O)cc(F)c1 N1(C(CCOC(C)C)=O)CCC(O)(CNC(C2C3CCC2(c2ccco2)C3)=O)C1 C1(C#CC(=O)N(CC(C)CNC(=O)CC2(C)CCCC2)C)(CC)COC1 CC1ON=C(C(=O)N2CCC(NC(c3coc(C(F)F)n3)=O)CC(O)C2)C1C N1(C(CCNc2cccc(OC)c2)=O)CCC2(CCCN2C(=O)CCCCCl)C1 C1(C(N(CCCNC(C(N2CCOCC2)C)=O)C)=O)CCCCCC1(F)F Cc1ccc(CC(=O)NC(CC(=O)NC2(C(N)=O)CC2)C2CC2)cn1 C#CCC(CC(F)F)C(=O)NCC(F)(C(=O)N1CC=CC(O)C1)C(C)C C(=O)(CC(C(C)CC)NC(C1(OC)CCOC1)=O)NCCCCCCC=C C1(C(N2CCC(C)(CCC)C2)=O)CCCCN(C(c2snnc2C)=O)C1 Cc1cc(C#N)ccc1-c1nc(C(=O)NCCc2cnc[nH]2)c(C)s1 N1(C(CNC(CC(C)C)=O)=O)CC2CC(C(N3CCCC(O)(CO)C3)=O)CC2C1 c1(C(N2CC=CC2Cn2cc(-c3cn[nH]c3)nn2)=O)c[nH]c2cc(Cl)ccc12 Cc1c(F)ccc(N)c1C(=O)NCC(C)CNC(C1CCCN(CC(F)F)C1)=O c1(C(N(CCCNC(=O)CC2CC(n3cnnc3)C2)C)=O)csc(C2CC2)n1 C(CCC(C)NC(=O)C(n1ccc(Br)n1)C)NC(CN(C(=O)OC)C)=O C1(NC(c2cc(C)cc(O)n2)=O)CC2CC1CN(C(c1cc3occc3s1)=O)C2 Cc1cc(=NC2CC(C(N)=O)C2)[nH]c(N2CCC(C)(CN3CCCCC3)C2)n1 CCCC(CCCO)C(=O)NC1CCN(C(=O)C(C(C)C)c2ccccc2)C1 c1(C(=O)NC(CNC(CCCC=C)=O)(C)C)noc2c1CC(C)CC2 CC1(C(=O)NCC2CCC2NC(c2cnoc2C2CCC2)=O)CC(F)C1 N1(C(CNC(c2n(C)ncc2)=O)=O)CCSC2CCCC12 c1(C(C)NC(=O)Sc2ncc(C(F)(F)F)cn2)ccc(Cl)c(Cl)c1 Cc1cc(C)n2cnc(C(N3CCC(NC(C4(C)CCCOC4)=O)CC3)=O)c2n1 N1(C(c2cc(C)on2)=O)CCC(C(=O)NCC(=O)NC(C)(C)C)C12CC2 c1(SC)ccc(C=CC(=O)NC(C)CCNC(=O)Cc2ccc(C#N)cc2)cc1 c1(CC)[nH]nc(C(=O)NC2C3CN(C(C4(C)CC(C)C4)=O)CC23)c1[N+](=O)[O-] c1(C(C)OC)nc(C(=O)NCCCC2(O)CCC2)cs1 c1(C(N2CC(n3cc(NC(C4CC5CCC45)=O)cn3)C2)=O)ccc(O)cc1 N1(C(CC(C)OC)=O)CCOC2(CCN(c3ncc(C#N)cc3Br)CC2)C1 c1(NC(N2CCCC(CCC)C2)=O)cc(COC)ccc1CO C1(C(=O)NC2(C)CCN(C(C(c3cccnc3)C)=O)CC2)CCCCC1C1CC1 C1(C(C(=O)N2CCC2C(N)=O)NC(=O)C(c2ccccc2)=O)CCCCC1 c1(CC(C(=O)NCCN(C(=O)Cc2ccon2)CC)O)ccc(OC)cc1 C(CC(C)CC)(C(=O)N1CC(C2=NOCC2)C1)NC(C(=O)NCC)=O c1(CN2CCC(CC(=O)NCc3n(C)nnc3)C2)cc(F)cc(Cl)c1O O=C(CC(C(F)F)n1cccn1)NC1CC2(C1)CC(NC(C13CCC1C3)=O)C2 C#CCC(CC(=O)NCCOC)NC(C1CCCC(=O)CC1)=O C(=O)(N1OC2C=CC1CC2)C1N(C(C(C(C)(C)C)CO)=O)CC(O)CC1 Cn1c(C(=O)NS(=O)(=O)CC23CCCC2C3)cnc1C(F)(F)F C1(NC(CCCC(CC)C)=O)CCC2(CCCN2C(c2nccnc2C)=O)CC1 CS(=O)(=O)C1(C(=O)NCC2CN(C(=O)C3=C(Cl)CC3)C2)CC1 CC(=O)C(C)(C)CC(=O)NCC(O)C(N1CCCC1(CO)CO)=O C12(CNC(CCc3cncc(C)c3)=O)CC(NC(=O)CC3=CCCC3)(C1)C(C)O2 C1(C)(C(=O)NCC2(NC(CCc3ccc(C)s3)=O)CC2)CCCCO1 C(=O)(C(CC)C(C)O)NC(CNC(c1n(CCC)ncc1)=O)C CCCCCC(C)(C)C(=O)Nc1cc(F)c(Cl)cc1Br N1(C(c2c(C)ncc(Cl)c2)=O)CC2CCCC2(NC(=O)C=C2CCC(C)C2)C1 CC1COCCC1CNC(C12CC(C1)C(C)O2)=O CCCC(C(N)=O)NC(=O)C(CCC1CC1)NC(=O)CN(C)C(C)=O NS(=O)(=O)c1cccc2c1CCN(N1CCCC1C1CCCCC1)C2 N1(C(c2cc(C#N)oc2)=O)CCCCC(NC(=O)CNC(=O)C(F)(F)F)C1 c1(C(=O)NC2C(CNC(c3cnc(C)[nH]3)=O)C2)cncc(C(F)(F)F)n1 n1(CC)cc(CC(=O)NCC(=O)NCC(=O)NC2(CN(C)C)CC2)cn1 N1(Cc2nc(CC)on2)CC(NC(c2conc2C(F)(F)F)=O)CCC1C C(C(=O)NC(C(=O)C(COCCSC)=O)C1CC1)(C1CCCC1)NOC N1(C(c2c(C)cc(Br)o2)=O)CCCC(C)C1CCNC(c1ccc(C#N)[nH]1)=O c1(C(N2CC3C(C(=O)NCCC(F)(F)F)(C3)C2)=O)cc(F)ccc1I c1(C(=O)NC(C2CCN(C(Cn3ccc(C)n3)=O)C2)C)cc2c(F)cccc2[nH]1 c1(C(N2CC=C(CNC(C3C=CCCC3)=O)CC2)=O)n[nH]c2c1CSCC2 c1(OC)cc(NC(C(C2CCN(C)CC2C)NC(=O)OC(C)(C)C)=O)nc(Br)c1 c1(CN(CCC#C)C(=O)CNC(C)CC)ccncc1 N1(C(c2c(C)cc(O)nc2)=O)CCC2CCCC12C(=O)N(CCCN(C)C)C N1(C(CCCc2n[nH]c(=N)s2)=O)CCCC(F)(CNC(C2CC(Cl)(Cl)C2)=O)C1 CCC(CC(=O)N1CC2CC1CN(C(=O)C(C)SC)C2)C(C)C CC(CC(F)(F)F)C(=O)NCC1(C)CN(C(c2ccc(N=[N+]=[N-])cc2)=O)CCO1 c1(SC)nc(N(Cc2ccc(Br)cc2F)CC2(O)CCCNC2)c(Br)c(C)n1 CCC(CC(=O)NC1CC(CO)N(C(=O)CC2(C)OCCO2)C1)C(C)C CCCCC(C)C(=O)N1CCN(C(c2ccc(SCCCO)cc2)=O)C2CC12 c1(C(N2CC(CNC(CN(C(C)C)C)=O)C(C)C2)=O)cc(F)c(F)cc1F C1(C(C)C)CCN(C(c2cnc[nH]2)=O)C(CNC(C2CC2c2ccoc2)=O)C1 N1(C(c2c(CC)nc(C)s2)=O)CCN(C)C(CNC(=O)C(C)(C)c2ccns2)C1 C(C(=O)NC1(CO)CCN(C(=O)Cn2cc(C3CC3)nn2)C1)(C(C)C)SCC C12(CNC(=NCc3ccc(OC)cc3)NC3CC(SC)C3)CCC(C1)C(C)(C)O2 C#CC1(O)CN(C(C2CSCN2C(c2coc(C(C)C)n2)=O)=O)C1 C1(OC)CC2(C1)CC(NC(C1CN(C(=O)CSC(C)C)CC1C(C)C)=O)C2 N#Cc1c(Br)cccc1S(=O)(=O)Nc1cccc2c1ccn2CC(=O)O C12(CCSC1)N(C)C2=O.C1(CN(C(C)=O)C(C2CCC(=O)N2)=O)CCCOC1 C#CCCC(C(=O)N1CCC(C)(CCC)C1)NC(=O)C(C)O C#CC1(C(N2CC(O)(CCNC(=O)Cc3cnccc3C)C2)=O)CCCC1 c1(CC2(F)CN(C(C)=O)C2)cccc(O)c1.C12(C(=O)OC)CCC1N2.C(C)(C)(C)O n1(CC)nc(C)c(C(=O)NCCOC(C)(C)CNC(=O)CC(CC)OC(C)=O)c1C N1(C(C(C)=C2CC2)=O)CC(C)CC1C(=O)NCC(C)(C)C#N c1(NC(CN(C(=O)COC(C)(C)C)CCOC)=O)cnn2c1OCCC2 C(=O)(C1=CS(=O)(=O)c2ccccc21)NC1CN(C(CSCC)=O)C2(C1)CCOC2 C(=O)(C(F)(F)C1CC1)NC(CNC(CCN(CCCCC)C)=O)C N1(C(CCOCC#C)=O)CCN(C(C2CCCOC2C=C)=O)C(CCO)C1 C1(NC(c2c(OC)cccc2)=O)CC12CCN(C(=O)Cc1cc(C)no1)C2 C1(CC(C)C)CC(C(=O)NCC2(F)CN(C(C3CCCCCC3)=O)C2)CC(=O)N1 c1(CCC(=O)NC2C(NC(C(C=C)c3ccccc3)=O)COC2)ccnc(C)n1 Cc1ccn(C)c1C(=O)NCCc1cc(C(=O)NC2CCS(=O)(=O)C2)no1 S(=O)(=O)(c1cccc(=NCc2ccco2)[nH]1)NCc1scc(C(N)=O)n1 C=CC1(CC(N2CCC(COCC)CC2)=O)CN(C(=O)CC2CC2)C1 Cc1ccc2c(CNC(=O)C(N3CCC(NC(C)C)CC3)=O)ccc(O)c2n1 C1(CNC(C(C)=C2CC2)=O)CCCCCN1C(c1ccc(OC(F)F)cc1)=O C(C)(N=c1nc2scnc2c(NCc2ccc(Cl)c(Cl)c2C)[nH]1)c1nnc(C)s1 N1(C(C2CN(C)C2)=O)CC2(C=C(C(=O)N3CCCCCC3)CO2)C1 N1(C(C(C)SCCCC)=O)CCC2CC2(C(N2CC(OCC(N)=O)C2)=O)CC1 C(=O)(CC1=CCCCC1)N1CCC(CN(C(C(C)N(C)C)=O)C)C1 C(=O)(CCCC(N)=O)N1CC(O)(CN(C(C(CC)C)=O)Cc2ccccc2)C1 C(=O)(CS(=O)(=O)C1CC1)NCC1(CNC(C(C2CCCOC2)OC)=O)CCC1 CCC(CC)CCC(=O)N1C(C)C2CC1C2NC(=O)CC1(O)CCC1 C12(NC(=O)Cc3ccc(CO)cc3)CCCC1N(c1nc(Cl)ncc1F)CC2 C1(CNC(C2ON=C(C(C)C)C2)=O)(NC(=O)C=CCO)CC2CCC1CC2 N1(C(C(CC)SC)=O)CCc2sccc2C1CNC(=O)Cc1ccnc(Cl)c1F C(=O)(CCCC(F)(F)CO)N1CCC(CCNC(c2c(C)cc(C)[nH]2)=O)C1 c1(C(N(CC(CN(C(=O)COCCF)C)O)C)=O)cc2n(c1)CCC2 C(=O)(C1CCc2ccccc21)N1CC2CC(NC(c3c(Cl)ncc(C)c3)=O)C2C1 C(c1ccc(Br)o1)=CC(=O)OC1CC=CCC1 C(=O)(CCCNC(N)=O)N(CC(CC)NC(C1(CF)CC1(F)F)=O)C CCCCC(O)C(=O)N1CCOC(C(C)NC(=O)CNc2ccc(Cl)cc2)C1 C1(NC(c2cn(C)c(=O)n2C)=O)CCCCC12CCN(c1cncc(Cl)n1)CC2 N1(C(C(N2CCOCC2)C)=O)CCOCC1CC(=O)Nc1cccc(CO)c1 CC(C(=O)NCCCOCCNC(C1CSC1)=O)NC(N)=O S(=O)(=O)(c1nc(N(CC(C2CCCCC2)O)C)ccc1Br)NCC1CN(C)C1 C1(C2(O)CCN(C(C3CCN3C(C)(C)C)=O)CC2)(NC(C=CCCC)=O)CC1 c1(C(N2CCN(C(N3CCN(C(N(C)C)=O)CC3)=O)CC2)=O)cc(Cl)ccc1I CCCCC(CC)C(=O)NC12CC(CNC(=O)C3CC3)(C1)OC2(C)C N1(C(C(CSC)C)=O)CCC(CNC(C2CCCN2C)=O)C(F)(F)CC1 C1(C(=O)NCCN(C(C)C)C)CC(O)CN1C(=O)Cc1cn(C)nn1 N1(C(c2ccc(CN3CC(C)C(C)C3)cc2)=O)CC(S(=O)(=O)NCCO)C1 CC1CC(C(=O)NCC(=C2CN(C(=O)CCN3CCCCC3)C2)F)CC(C)C1 CCCC(C#N)C(=O)N1CC(O)CC1CNC(=O)C(C1CCCC1)OCC N1(C(C(C(C)O)N(C)C)=O)CCCCCC1CNC(=O)Cc1ccc(Cl)s1 S(=O)(=O)(CCC(=O)NC1CN(C(=O)CC2CNC(=O)C2)CC1OC)NC C1(C(N2CCN(CC(C)NC(c3n(C=C)ncc3)=O)CC2)=O)CC2C(C1)C2(F)F N1(C(C2(CSC)CC(F)(F)C2)=O)CCCC(CO)(NC(=O)C(C)n2cncn2)C1 c1(C(=O)NC(C2CCN(C(c3c(CC)cco3)=O)C2)C)cc(CC)c(=O)n(C)c1 C1(CCOC)(NC(=O)CC2C=CCC2)CCN(C(C2(C)CCCO2)=O)C1 C(CN=C(NCC1CCC1)NC1CCC1(C)C)c1cc(C)sc1C S(=O)(=O)(c1cc2sc(=NC(C)C3CCC3)[nH]c2cc1Cl)N1CCC(C(C)C)CC1 N1(C(c2c(C)occ2)=O)CCC(C2CC(NC(=O)Cc3cc(F)ccc3F)C2)C1 c1(OC)nc(C)ccc1C(=O)N(CCCCCCNC(C1CCCN1C)=O)C c1(NCC)ccc(C)cc1C(N1CC(NC(=O)CS(=O)CC)CC(F)C1)=O CC(C)CC(C)(CNC(C1CC12CC(C)(C)C2)=O)NC(c1cn2c(n1)SCC2)=O N1(C(c2cccc(OC)c2O)=O)CCC2C1CCN2C(=O)CNC(=O)O C(C(C)C(C)C(=O)N(CC(=O)NCC(C)(C)c1cccs1)C(C)(C)C)OC CCCCC(C(=O)NC1CCN(C)C(=O)C1)NC(c1cnns1)=O Cc1cccc(C)c1C(=O)NC(C1CCN(C(c2csc(C)c2C)=O)C1)C c1(-n2cc(CN(C3CCC3)C)nn2)cc(S(N)(=O)=O)ccc1Cl CC1=C(C)CN(c2nnc(-c3ccc(OC(F)F)cc3)n2C)CC1 C1(CNC(C(CC#C)O)=O)CCCN(C(c2c(C)nsc2Br)=O)CC1 c1(C(=O)NCC2(C)CCN(C(C3CCN(C)C3)=O)C2)cc(O)nc2c1CCCC2 c1(SCC(=O)N(CC(C)NC(c2ccc(C(=O)OC)o2)=O)C)cc2c(s1)CCC2 C12(CO)CCCN(C1)C(=O)OC2.n1(COC)nccc1C(=O)OC(C)(C)C C(c1ccccc1)=CCC(=O)NCC(C(=O)NC(C#C)CC1CC1)C Cc1cccc(C(F)C(=O)NC2CC(C(C)NC(C3(C4CC4)CC3)=O)C2)c1 CCC(CNC(=O)C(C)C(C)NC(=O)Cc1nonc1C)CC(C)C c1(CN2CC(C(=O)NC)C(O)CC2)ccc(OC)c(O)c1Cl C1(C(C)C)CCN(C)CC1.c1(C(=O)N)cc(-c2ccccc2)nn1C.C=C1CC(C)C1 C(=O)(C(F)CC(C)(C)OC)NCC(C(=O)Nc1cnc(F)cc1C)OC c1(OC)cccnc1C(F)(F)C(=O)N(CC(C1CC1(F)F)=O)C c1(C(C)NC(c2n(CC(=C)C)nnn2)c2ocnc2CC)ccc2c(c1)CCC2 C(C(=O)NNC(=O)OCCO)C1CC(OCc2ccc(OC)cc2)C1 c1(C(=O)NC2CCCCN(C(COCCOCC#C)=O)C2)cc(C)c(Cl)cc1F N1(C(c2ncn(C)c2C(F)(F)F)=O)CC2CCN(C(=O)CSCC(=O)O)C2C1 C#CCCC(C(=O)NC1(CCF)CC(O)C1)NC(=O)CCC(C)N(C)C C1(C2(C=C)CCC2)(C(N2CC(C=C)C(NC(=O)C(C)(C)OC)C2)=O)CCC1 c1(OC(C(=O)NCCC(CNC(C(CC)C)=O)O)(C)C)cccc(C(C)C)c1 C1(C(=O)NC(CNC(C(C)SCC)=O)(CC)CC)CCC2(CCC2)C1 c1(CNC(=O)Cc2ccoc2)cc(Cl)n(C)n1.C1(OCC)CC(C2CCCO2)C1 N1(C(COC)(C)C)CCN(C(=NCCSC)NCc2cnc3n2CCOC3)CC1 n1(C2CN(C(=O)OC(C)(C)C)C2)cc(CN(CCCO)C2CC2)nn1 C1(C(=O)NCC2(CCNC(C(C)NC(C)=O)=O)CC2)CCCC(F)(F)C1 CC1CN(C(=O)CC(O)CN(C)C)CCN(C(C2CCCCC2N=[N+]=[N-])=O)C1 C(CCC(CCC)NC(=O)C=C(Cl)Cl)OCCCCCCC.C1(=O)C(CCC)N1 N1(C(c2ncn(C(C)C)c2)=O)CCN(C(C2CC(O)CN2C)=O)CC2(CC2)C1 C=CC(C)(O)CC(=O)N(CCC(C(C)(C)C)NC(=O)C=Cc1ccc(C)cc1)C C1(NC(C(C)OCC=C)=O)(CNC(=O)C=Cc2cnc[nH]2)CCC(C)(C)CC1 Cc1cc(C(=O)NC2(C)CC(NC(c3coc(C(F)F)c3)=O)C2)n2ncnc2n1 C1(N(C(=O)COc2ccccc2)C)CCCN(C(C2(C)CCC3CC3C2)=O)CC1 c1(OC(C)C)ccccc1CC(=O)NCC1CCC(c2ccccc2)C1 C1(CNC(CP(C)(C)=O)=O)CN(C(=O)Cc2ccc(O)cc2Cl)CC1(C)C CC(C)(C)C(C(=O)N1CCCC(NC(=O)C=CC2CC2)CC1)C1CCCC1 C1(NC(C(C)NC(c2ccco2)=O)=O)CCC(NC(C2CN(C)C2)=O)C1 c1(CN2CCC(CNC(c3cccnc3)=O)C2)cccc2cccnc12 C#Cc1ccc(OCC(=O)N(CCNC(=O)CCc2cnc[nH]2)CCOC)cc1 C1(C(N(CC)CC2CCCCO2)=O)CC2CC2N1C(c1cc(CO)[nH]n1)=O c1(N(CC(=O)N(CC)CC)C)nc2ccsc2c(=NCc2cncc(Br)c2)[nH]1 C(=O)(C(C)(O)C(F)(F)F)NC1CN(C(c2c(OCCC)cccc2)=O)C1 c1(C(=O)NC(CC)(C)CNC(=O)CC=C(Cl)Cl)cnn2c(OC)cccc12 Cc1cc(C(=O)NC2(C(=O)NC3CCCC34CC4)CC2(C)C)ccn1 C1(CC)C=CCN(C(=O)CC(C)(C)N(C(=O)C(O)C(C)C)C)C1 N1(C(=O)COC2CCOCC2)CCC2CC1CN(C(C1(CCF)CCC1)=O)C2 C1(C(N2CC(NC(CCCC(=C)C)=O)C(C)(C)CC2)=O)CCN(S(N)(=O)=O)CC1 CC1=CCC(NC(=O)CCC2CCCN2C(=O)C#CC2CC2)CC1 N1(C(=O)NCC2C3COCC23)CCCc2c(F)c(F)cc(F)c21 c1(COC)ccc(C(=O)N(CCCCN(C(=O)CN2CC3CC3C2)C)C)cc1 Cc1ccc(-c2cc(C(=O)NCCCC(C)NC(c3cncs3)=O)no2)c(C)c1 N1(CCc2cccc(C(C)(C)C)c2)C(=O)NC(c2nccs2)C1=O N1(C(C(=O)NC(CC#C)CC)=O)CCCC(O)(C(C)C)C1 C12(C(=O)NCC(C)NC(c3c(OC)noc3C)=O)CC3CC(F)(C1)CC(F)(C3)C2 C(=O)(C1=CN=C2N=CNN2C1)N1CCC(CNC(C2CC=CCC2)=O)C1 N1(C(c2cnc(C(C)C)[nH]2)=O)CCC(C(C)NC(=O)C(O)CC2CC2)CC1 c1(C(N2CC(C(C(=O)NC(COCCOC)C)OC)C2)=O)ncnn1C1CC1 C1(C(=O)NCC(C)(CO)NC(C2(C(F)(F)F)CC(F)(F)C2)=O)CCCCCC1 CCCCC(F)C(=O)NC(CSC)C(=O)N(C1(c2cc[nH]n2)CC1)C c1(NC(CCC)C)ncc2ccccn12.C1(=O)CN(C)CCOCCN1C C1(NC(c2c(C)cc(C)s2)=O)CS(=O)(=O)CC1NC(=O)CN1CC=CC1 Cc1coc(C2CC2)c1C(N1CC(NC(C2NC(=O)OC2C)=O)C(C)C1)=O CCC(F)(F)CC(=O)NC(C)(CNC(=O)CC1CCC(C)CC1)C1CC1 C1(C(N2C(C)CC(CNC(=O)Cc3nnc(O)s3)C2)=O)C(C)(C)CCCC1(C)C C1(C(=O)NCc2cccc(C)c2)CC2(CCN1C(=O)C(O)CC1CCCC1)CC2 C1(C)(C(=O)NCCCC2(NC(C3CC(CSC)C3)=O)CC2)C=CCC1 c1(NC(C2CCCN(C(C(=O)NCC#C)C)C2)=O)csc2cncn12 C1(NC(C2C(OC)C2)=O)CCN(C(c2ccc(C(F)F)o2)=O)CC1(C)C n1(CC(=O)N(C2CCN(C(c3n[nH]cc3C)=O)C2)CCC)cc2ncccc2n1 CCC(C)CCCC(=O)N(CCNC(C1OCC2CCCC1C2)=O)CC c1(OC)ccc(NC(C2(NC(=O)CNC(C3CC3C)=O)CC(O)C2)=O)cc1 C1(NC(Cc2cc(C)no2)=O)CCCC(N(C(=O)CCCF)C)C1 CC(C)C(C)C(C)CC(=O)N1CCN(C(=O)CCC[N+](=O)[O-])CC1C(C)C CCCCC(C(=O)NC(CC(=O)NCCCCC1CC1)C(C)(C)C)C(C)C C1(C(N(C2CCN(C(c3cnc(C)c(N)c3)=O)C2)CC)=O)CC2CC(C1)C(=O)N2 C(=O)(CCCN(C)C(C1CCCO1)=O)NC(c1ncc[nH]1)C C(=O)(C1CCCc2nn(C)cc21)N(CCCNC(CCSCC)=O)C C1(C(=O)NCC2CN(C(C#CC3(C)CC3)=O)CC2O)Cc2cccc(F)c2O1 c1(C(CO)NC(C2(C)CN(C(C3CC3C3CC3)=O)C2)=O)cccc(F)c1 NS(=O)(=O)c1cc(C(=O)NC2CCC2CNC(C2(CO)CCC2)=O)cs1 c1(C(=O)NCC=CCNC(C(CN(C)C)(C)C)=O)c(N)c(F)cc(F)c1F c1(C(N2C(CNC(C(C)O)=O)C=CC2)=O)ccc2ccccc2c1F N1(C(C(=CC2CCCC2)C)=O)CC2CC2(CNC(c2nc(C)oc2C)=O)C1 N1(C(C2(C)C(C)C2)=O)CCC2(C(=O)NC(c3ccc(O)cc3)CO)CC2C1 C1(OC)CN(C)C(C)(C(=O)N(C(CNC(c2nc(Cl)sc2C)=O)C2CC2)C)C1 c1(OCC=C)ccc(C(=O)NCCC(C)NC(=O)OC(C)(C)C)cc1 c1(CC(N2CC(OCCNC(C(CC)OC)=O)C2)=O)cc(Cl)n(C)n1 Cc1ccc(CN(C=O)Cc2c(C)nn(C)c2-n2cccn2)cc1Br C1(CC(=O)NC(CNC(Cc2c(C)cccc2)=O)C)Cc2ccccc2O1 N1(C(C2CC(CNC(C(CC)=CC)=O)C2)=O)CCCCC1C(C)(C)C C12(CC(=O)NCc3cc(C)c(C)o3)CCC1CN(C(c1c[nH]c(C#N)c1)=O)C2 c1(COC)cccc(C(=O)NCC#CCNC(c2ccncc2Cl)=O)c1C c1(OC)cccc2c1CN(C(C1Cc3cccc(F)c3O1)=O)CC(C)(C)O2 c1(NC2CCC(N(C(C(C(C)O)(F)F)=O)C)CC2)ncnc2c1CCC2 c1(C(N(C)CCNC(=O)CCc2ccc(F)nc2)=O)cccc2c(C#N)c[nH]c12 c1(C(=O)NCC(CO)NC(C2N(CCC)CCC2)=O)cnn(C)c1N C(C(C)CN=c1[nH]nc(C(C)(C)C)s1)NC(COC(CC)C)=O C=CCCCCCC(=O)N1CC(=O)NCC1C(=O)NCCC(C)C(C)C N1(CC(=O)N(C2CCCC2)CCNC(c2cocc2C(N)=O)=O)CCSCC1 c1(C(=O)NC(c2nc(N3CCC(N(C)C)C(C)(C)C3)sn2)C)ccc2nn[nH]c2n1 N1(C(C2CN(CC(C)C)C(=O)C2)=O)CCCCC(NC(=O)C(F)F)C1 c1(C(=O)NCC23C(CN(C(C(C)OC)=O)C2)C3)c(C)ccc(C)c1C CCCCC(C(=O)NC1CN(C(c2ccc(CC)s2)=O)CCC1C)C(C)C C1(C(=O)NCC2(S(N)(=O)=O)CC2)(NC(CC(C)C)=O)CCc2cc(Br)ccc2C1 CC(C)C(F)C(=O)NCC(C)(C)CNC(=O)Cc1ccc(Cl)cc1 C12(CNC(CSc3nc(C)[nH]n3)=O)CN(C(=O)CN(C)C(N)=O)CC1CCO2 C1(NC(Cc2c(C)n(C)nc2)=O)CCN(C(c2cc(N)ccn2)=O)CCC1CO C1(C(N2C3CN(C(C(C)C(=O)OC(C)(C)C)=O)C(C3)C2)=O)CN2CCN1CC2C C(=O)(CS(=O)(=O)CCO)N(C1CCCCC1)CCNC(C1C(CC)CCO1)=O N1(C(Cc2nc(C)[nH]n2)=O)CCC(F)(F)C(C(=O)CCNc2ccccc2Cl)C1 Cc1ccc(F)c(OCC(N2CCCOC(CNC(c3ccsc3C)=O)C2)=O)c1 N1(C(C(CC)(C)OC)=O)CCOC2(CCC(NC(c3cc(OC)ns3)=O)CC2)C1 c1(C(N2CCCC(N(C(=O)CC3(COC)CC3)CC)C2)=O)c[nH]c2ncccc12 CCS(=O)CC(=O)N1CCCCC1C1CCN(C(C2CC2c2ccccc2)=O)C1 c1(C(N2CC(C(=O)Nc3c(C(N)=O)cccc3)SCC2)=O)cccc(O)c1O c1(C(=O)NC2CC(CCNC(Cc3c(C)n[nH]c3)=O)C2)ccc2c(c1)C(=O)OC2 c1(OC)cc(C(N2CC(CNC(c3ncnn3C)=O)CC2C)=O)nn1C O(NC(=O)C=Cc1nccs1)CC(=O)NCCNC(N)=O C1(CC(N2C(CNC(=O)CN(C3CCSC3)C)CC3CC23)=O)(OC)CCCCC1 N1(c2n(CCN(C(=O)OC)C)nnn2)CCOc2ccc(C)cc2C1 N1(C(C2(C)CCC2)=O)CC2CN(C(c3ccc(CC#N)cc3)=O)CC2C1 C1(C(N(C2CC3(CCC3)C2)C)=O)N(C(C2CC2C2(C)COC2)=O)CCCC1(C)C C(=O)(C1COCc2ccccc21)NCCC1(CNC(c2cc(C)oc2C)=O)CC1 c1(C(=O)NCCC(C(C)C)NC(CC(CCC)O)=O)c(O)nc(=O)n2c1CCC2 n1(CCC(=O)NCCn2nccn2)cc(-c2ccc(C3CC3)s2)nn1 C1(NC(Cn2c(C)ccn2)=O)CCN(C(=O)CC(O)CN(C)C)CC(C)(C)C1 C(C)(C)(CC(=O)NCC1(F)CN(C(=O)CSc2cccc(Cl)c2)C1)N(C)C CC1(C(N2CC(O)C(O)C2)=O)CCN(Cc2ccc(Cl)nn2)CC1 CCCC(CC)CCC(=O)NC1(C(=O)NCc2cnn(C)c2)CCCC1 C12(CNC(C3C(=C)CC3)=O)CCCC1N(C(C1CC=CC1)=O)CCC2 C1(CCNC(C(c2cccc(Cl)c2)(C)C)=O)COCCN1CCOCC(F)(F)F Cc1cc(=NC2CCN(CC(N)=O)CC2)[nH]c(N2CC(C)OCC(C)(C)C2)n1 C1(C)(CNC(n2cc(COCC(=O)O)nn2)C)CCCS1(=O)=O C1(NC(c2c(C)nc(C3CC3)[nH]2)=O)CCN(C(c2c(C)nc(C)n2O)=O)C1(C)C c1(CC)ccc(C)cc1C(N1CC(CCCCNC(=O)Cc2scnc2C)C1)=O c1(CC(N2CC3C(NC(C4C(F)(C(=O)OC)C4)=O)C3C2)=O)ncn2c1CCCC2 c1(C(=O)NCC(C)(C)NC(C(C)SC)=O)cc(C)c2ncccc2c1C c1(C(=O)NC2CN(C(C(CC)F)=O)CC2F)cc(S(=O)(=O)NC2CCC2)c[nH]1 c1(Sc2ccc(CC(=O)OC(F)(F)C(F)F)nc2)cccc(F)n1 N1(C(c2ncc(C(=O)OC)s2)C(=O)NCC(F)F)CCC(C2CCOCC2)C1 c1(C(C(=O)NC2(C=C)CC2)N(C(=O)OC(C)(C)C)CC)ccccc1F C1(NC(c2c(CC)cccc2)=O)CCN(C(=O)CC2(C)CC2(Cl)Cl)CC1F N1(C(C(CCC)C(C)C)=O)CCC2CN(C(C3CC(C)OC3C)=O)CC2CC1 C(C)(C(CCC(=O)O)CCCC(=O)O)NC(CC(=O)OC)C(=O)N1CCNCC1 CCC(C)(CC(=O)N1CCC(CN(C)C(c2cc(C)no2)=O)CC1)C(=O)OC N1(C(Cc2cc(C)on2)=O)CCCC(CNC(=O)CC2CC3(CC3)CO2)CC1 N1(C(Cn2nc(C)c(Cl)c2)=O)C2CCCC1CN(C(c1cc(=O)cc[nH]1)=O)C2 c1(C(=O)NC2CC(N(C(CCC=CC(C)C)=O)C)C2)cc(Cl)c(Br)[nH]1 C(=O)(C(O)CN(C)C)NCCN(C(=O)C(n1cnnn1)C1CC1)CCOC C1(C(=O)NCC(C(C)C)(C)NC(=O)C2=CCCCO2)CCCC(F)(F)C1 C1(CC)CC12CCOC2.c1(CC(=O)N(C(C2CCC2)C)C(=O)OC)ccoc1 N1(C(c2cc(OC)ncc2Cl)C(=O)NCCCC)CCCC(O)(COC)CC1 C(C(C(C)(C)C)NC(=O)NC(Cc1ccnnc1)=O)NC(=O)OC(C)(C)C C1(C(=O)NC2(CNC(C(NC(C)=O)=Cc3cccs3)=O)CCC2)CCCC(=O)O1 C1(CC(=O)N(C2CCC(NC(c3sccc3C3CC3)=O)CC2)C)CCCCCO1 CC1CC(NC(c2cnn(CC(F)(F)F)c2)=O)CN(C(C2CCCC2)=O)C1 c1(C(=O)NC2C(NC(C(c3c(C)noc3C)C)=O)COCC2)cccc(Cl)c1F N1(C(CCC)=O)CCC(C(F)CNC(c2ncoc2Br)=O)CC1 N1(C(c2c(C)ccn2C)=O)CCc2c(C(=O)NCC3(C)CCCC3)cccc2C1 N1(C(C2(CC)CCC2)=O)CCCCC(N(C)C(c2cc(C)cs2)=O)C1 C1(NC(C2C(C=C)C2)=O)CCC(C)(CNC(c2cccnc2N(C)C)=O)CC1 C1(CC)(CO)CN(C(=O)C(F)=C(C)C)C1 c1(C(=O)NCC2(NC(CCN(CCCCOC)C)=O)CCC2)n[nH]cc1[N+](=O)[O-] c1(OCOC)ccc(CNC2CN(C(c3ccsc3C)=O)CC2C)cc1 c1(OCC)cc(C(=O)NC(C)(CNC(=O)C(C2CCCC2)OC)CC)[nH]n1 c1(CCC)n[nH]cc1C(=O)NCc1cc(C(=O)N(CCCO)CC(C)C)cs1 n1(CC(=O)NC2CN(C(C(CC)F)=O)CC(C)C2)c(C)nc2ccccc2c1=O c1(CC)nn(C)c(C(N2CCC(NC(c3ccc(Cl)c(Cl)n3)=O)C(F)C2)=O)c1Cl C1(C2(C(=O)N(c3ccsn3)Cc3ccsc3Br)CC2)CCCN1CCO c1(CC(=O)Nc2cccc(Cl)c2Cl)ccc(-c2nccnc2OC(F)F)c(F)c1 c1(NC(=O)CC(F)(F)F)cccc2c(Cl)c[nH]c12 Cc1nnc2n1CC(C(N1CCC(CNC(c3csc4nccn34)=O)CC1)=O)C2 C1(CNC(=O)CC2C=CCC2)CC2CCCCC2N1C(c1ccnn1C(F)F)=O c1(C(N2CCN(CC3C(C)C=C(C)CC3)CC2)=O)occc1C1=CCNCC1 c1(C(=O)OCC2CC2)cc(F)cc(F)c1O.N12CCCC(C1=O)NC(=O)C2 c1(C(N2CC(OCCNC(CNC(C)=O)=O)C2)=O)c(C)csc1Cl c1(C(=O)NC2CCN(C(c3cnn(C)c3Br)=O)C2)ccc2c(c1)CCC=C2 c1(C(C)C)cc(C(=O)NC(C(C)NC(c2cccc(Cl)c2)=O)C(C)C)ccc1F c1(C(=O)NCC2CC(NC(C3(C)CCCCO3)=O)C2)cc(C(F)(F)F)ccc1O Cc1cc(=O)c(C(N2CCC3(C(N4CCC(C(N)=O)C4)=O)CC3C2)=O)c[nH]1 c1(CN2CCC(NC(c3cnco3)C)C2C)cccc([N+](=O)[O-])c1 C1(C(N2CCOC(C(F)(F)F)C2)=O)CN(Cc2c(Br)cccc2Br)CCC1(F)F c1(C(=O)NCC(C)N(C(=O)CC2CC2c2cnc[nH]2)C)ccccc1CC#N CC1CCCCC1(C)C(N1CC(C)(NC(=O)CCC(=O)c2cccc(N)c2)C1)=O N1(C(c2n[nH]c(C(C)C)c2Br)=O)CC2CC(NC(=O)CC3(N(C)C)CC3)C1C2 c1(OCC(=O)NC2C(NC(CCCC)=O)CCC2)ccc(C)cc1OC(C)=O c1(OC)cc(F)ccc1CC1CCCN(C(c2cnccc2N(C)C)=O)CC1 C1(NC(COC(CC)CC)=O)CCN(C(=O)CN2CC(C)C2)CCC1CO N1(C(C2CC(C)(F)C2)=O)CCOC(CCCNC(c2n[nH]cc2C(F)(F)F)=O)C1 N1(C(C(C(C)C)SCC)=O)CCCCCC(NC(c2cn(C3CCC3)nn2)=O)C1 C1(CC)CCCC(C(C(=O)NCCSC)N(c2cc(C(N)=O)ncn2)C)C1 Cc1nccc(C(N2CCC(NC(=O)C=CCCC(C)C)C(C)C2)=O)c1O C1(C(N2CCC2CN2CC(CC(C(=O)OCC)F)C2)=O)C2CC3C(C2)C13 C=CCC(C)(C(F)F)NC(=O)CC1CC(NC(=O)C(C)CC=CC)C1 c1(C(=O)NC(C)CNC(c2cnn(CC(F)F)n2)=O)c(F)ccc2c1OCC2 C(=O)(C(O)CC(F)F)NC1C(NC(c2ccc(CCC)[nH]2)=O)COCC1 c1(SCC)ccccc1C(=O)NCC(C(C)C)NC(=O)CCCC1CC1 Cc1nnc(C(=O)NCC2CC(F)(CNC(C3CCCC3O)=O)C2)s1 c1(OC)ccc(CC(=O)N(CCN(C(=O)Cc2csnn2)C)C(C)C)nc1 Cc1ccc(Br)c(F)c1C(N1CCOCC1C(=O)Nc1c(Cl)cccc1I)=O CC1N(C(C2COCCN(C(C3CC(=O)NC(C)C3)=O)C2)=O)CCCC12CCC2 c1(C(N)=O)ccc(C(N2CC(O)(CCNC(C3COCCO3)=O)C2)=O)[nH]1 O=C(Cn1cc(COCc2ccc(Cl)cc2)nn1)NNC(=O)c1ccco1 c1(CNC(=O)C(c2cccc(F)c2Br)F)cc2c(o1)CCCC2 C1(C(=O)NC2(CC=CC(=O)NC3C(C)CC3)CCC2)CNC(=O)N1 CCC(O)C(C)C(=O)N1CCC(CCNC(c2c(C(F)(F)F)noc2C)=O)C1 c1(CC(=O)NC2CCN(C(=O)CC3CCC(O)C3)C2)c[nH]c2cc(Br)ccc12 C(CCN=C(NCc1sccc1S(C)(=O)=O)NC1CSC(C)C1)SC c1(C(=O)NC2CC(CNC(c3cc(C)nnc3)=O)C2)cc2occc2[nH]1 c1(CSCC(=O)NCCN(C(=O)CC2CCCO2)CCC)ccc(Cl)cc1 CC1=C(C(=O)N2CC(N3CC(NC(=O)Cc4nc[nH]n4)CC3=O)C2)CCCO1 c1(C(=O)NC2C(NC(COCC(=C)C)=O)C2)ccncc1C(F)F c1(C(N2CC(CNC(c3nc(OC)oc3)=O)C(C)C2)=O)cc2cnn(C)c2s1 CCCC(C)(C)CC(=O)N1CC(NC(c2cc(C#N)cs2)=O)C(C)C1 c1(C(=O)C2CC2)cn(C(=O)NCC2CC(NC(C3(n4ccnn4)CC3)=O)C2)nn1 c1(C(=O)NC(C(C)NC(c2c(CCC)occ2)=O)C)onc(Br)c1C c1(SC)ccccc1NC(=O)C(CCN(C)C)NC(=O)CCc1ccn(C)n1 Cc1nc(C)c(CC(=O)NCC2(NC(c3c[nH]nc3Cl)=O)CCOC2)s1 CN1CCCCC1CC(N1CCCC1C(C)(C)CNC(=O)CSC(C)(C)C)=O C(CCN=c1[nH]cc2ccnc-2[nH]1)N(C(c1c(C)coc1C(C)C)=O)CCO C(=O)(C(C)(C)CCCF)N1CCN(C2CN(C(CN(C)CC)=O)C2)CC1 N1(C(=O)CCCCc2cnn[nH]2)CCCCC2(CCN(c3nccnc3F)C2)C1 Cc1c(Cl)ncc(F)c1COC(c1cncc(-c2cn[nH]c2)c1)=O c1(C(N2C(C3CCN(C(C4C(OC)CC4)=O)C3)CCC2)=O)[nH]c(C)cc1C C(=O)(C(O)(C(F)(F)F)C1CC1)NCCN(C(=O)CC1CN(C)CC1O)C C1(NC(C=NOC)=O)CCCC2CN(C(=O)CSCC(C)=O)CC12 c1(C(N2CCC(CN(C(=O)C(F)(F)c3ncc[nH]3)C)C2)=O)csc2ccccc12 C(=O)(C(C(C)C)C(C)C)NC1(C(=O)NC(C(=O)OC)C)CC1 C1(C(=O)NN(C(C)C)CCNC(C2(C(N)=O)CC2)=O)C2CCC12c1ccccc1 C1(CNC(=O)Cc2ccc(C(F)F)cc2)CN(C(=O)C(O)CC2CC2)CCCO1 C1(CC(=O)NCC(CC)(C)C)CCCN(C(=O)CC2CC=CC2)CC1 N#Cc1cnc(NC(C2CC23CN(C(C2CCCCO2)=O)C3)=O)c(Cl)c1 C(=O)(C(C(=O)NCC1CCCN1C(=O)CCCc1cccnc1)C(C)C)OCC c1(CC(N2CC(NC(C(CCSC)O)=O)(CO)C2)=O)c[nH]c2nccc(Cl)c12 N1(C(C2C(NC(CC(=O)NCC)=O)CCCC2)=O)CC2(COC(C)C2)C1 C=C1CCN(C(c2ccc(C)c(C)n2)=O)C(C(=O)NCCC(C)C(=O)OC)C1 C(=O)(C(CC1CCC1)OC)NC(CC)(C)C.C12(O)CN(C1)C(=O)C2F c1(NC(C(=O)NC(CC)CCOC)=O)cc(I)c(Br)cc1C c1(C(N2CC(CN(C(=O)Cc3ccoc3)C)OCC2)=O)cccc2c1OCCC2 Cc1cc(=O)n(C)cc1C(N1CCC(NC(=O)C2=COCCC2)C(C)(C)C1)=O Cc1cc(=NC(C)CCCO)[nH]c(=NCc2nnc3c(=O)[nH]ccn23)[nH]1 c1(C(N(C)CC2CCN(C(c3c(C)onc3)=O)C2)=O)nccc2c1CNC2=O c1(C(N2CCC(C)(CNC(=O)CCN3CCC3)C2)=O)ccc2cc(F)ccc2n1 C(C)(CO)(C(=O)NCCCC(C)(C)NC(=O)CSc1[nH]c(C)nc1C)NC(C)=O C1(C(N2CC3C(NC(C4CC5CCC(C4)O5)=O)(C3)C2)=O)CC2(C1)CC2(F)F Cc1cc(O)cc(O)c1C(=O)NC1(CNC(C2CCCCO2)=O)COC1 C1(NC(N(CCCNC(=O)CCC#N)CC)=O)(CO)CCC(F)(F)C1.C(C)(C)C C(=O)(C1=CCCCC1)N1CCC(N(C(c2ccc(CC)s2)=O)CC)CC1 CCC(C)(C)C(O)C(=O)NC1CCC12CN(C(c1cccc(OC)c1N)=O)C2 CCCS(=O)(=O)CC(=O)NCC1CC(OC)CN1C(=O)CCC(=O)OC C1(CC(=O)NCC(C)N(C)C(C2CC23CC(O)C3)=O)CCCOCC1 C(=O)(C(O)CC(C)C)N1CCC(C(C(=O)NCc2nc(C)c(Br)s2)C)CC1 N1(C(c2cn(CCC=C)nn2)=O)CCCC(NC(c2cccnc2S)=O)C1CC N1(C(Cn2cnc(C#N)n2)=O)CCC2CN(C(C3(c4cccs4)CC3)=O)C2C1 c1(C(N(C(C)CNC(=O)CC2(O)CCC2)CC)=O)ncnc2c1CCCC2 CC1CC(C(=O)N2CCN(C(c3cnn(CCO)c3)=O)CC2CC2CC2)=NO1 Cc1cocc1C(=O)NCC(C)CNC(c1c[nH]nc1-c1ccsc1)=O CC(CC(C)NC(c1c[nH]nc1I)=O)NC(=O)C(=O)N(C)C c1(C(=O)NC2CC(NC(CC3C=NN(C)C3=O)=O)C(O)C2)cccc(Cl)c1O C(=O)(C#CC(C)(C)CNC(C1(CC)CCCC1O)=O)N(C(C=C)C1CC1)C c1(CN2CCC(C)(NC(c3coc(C(F)F)c3)=O)CC2)c[nH]c2ccccc12 N1(C(c2ncn(CC)c2)=O)CCOC(C)(CNC(C2CCCCN2C(C)C)=O)C1 C1(C(N2C(CC(=O)OCC)CC2)=O)CN(C(c2ccoc2)=O)CC12CCC2 c1(OC)cc(C)ccc1CNc1nccc(N(C)CC2CC2(C)C)n1 CCC(CC)C(C)C(=O)NCC(C)(C)CNC(C1CCC(O)CN1C)=O c1(C(N2CC3C(CNC(=O)CC4(CO)CC4)C3C2)=O)cc2ncccc2o1 C1(C)(CNC(C(C=C)(F)F)=O)CCN(C(C2CC2c2ccnn2C)=O)CC1 C1(NC(NCc2n(CC)nnc2)=NCCN2CCOCC2)CCCCC12CCC2 C12(NC(C(C(=O)OCC)OC)=O)CCCC(NC(=O)CCCN(C)C)(C1)C2 C(=O)(C1=CC2C=CC(C1)C2)N(CCOCCC(N1CC(C#C)(F)C1)=O)C C1(C)(CC)CC(NC(=O)C=Cc2ccncn2)CN1C(=O)C=C1CCC1 c1(C2(NCC(CNC(=O)Cc3nc(C4CC4)cs3)OC)CC2)ccc(C)nc1 c1(C(N2C3CN(C(CN(C(C)=O)C)=O)CC2CC3)=O)cccc2cc(F)ccc12 c1(C(N2CC(CNC(C(CCOC)OC)=O)C2)=O)cc(Cl)c(F)cc1C N1(C(CC2(OC)CCCCC2)=O)CC(C)CCC1CNC(=O)CCC(F)(F)F C1(NC(C2CCC(C(=O)O)C2)=O)CNCC(F)(F)C1 N1(C(C)(C)CO)CCN(C(=O)C(C2(O)CCC2)NC(c2cccnc2)=O)CC1 c1(CC(=O)NCCC(Cn2cc(C(CC)CC)nn2)(F)F)ccc2occc2c1 c1(C(N2CCC(NC(c3coc(O)n3)=O)CC2)=O)c[nH]c2c(F)cccc12 c1(CCC(N2CCC(C(=O)NC3CCC(C(C)O)CC3)C2)=O)ccc(F)cc1Cl N1(C(C(C)NC(C)=O)=O)CCCC(O)(CCNC(C2(N(C)C)CCOCC2)=O)C1 N1(C(CSCCCC)=O)CC2(CCN(C(c3ncc(F)cn3)=O)CC2)CC1C CCCC(CC(=O)Nc1ccccc1C)NC(=O)CC1(COC)CC1 N1(Cc2ccc(CC)s2)CCC(=O)N(Cc2cccc3[nH]ccc23)C1=O c1(CCn2cc(CNC(=O)NC)nn2)cc(C)ccc1C O=C(C1CCSc2ccccc21)NC1CC(CNC(C23CCCC2OCC3)=O)C1 c1(N(C)C)cnccc1C(=O)NC1CC(F)(CNC(=O)CCc2nccn2C)C1 n1(CC(=C)C)nc(-c2cccc(N(C)CC)c2)nc1CC(C)C C1(C(=O)NC2CCN(C(CCC(C)N(C)C)=O)CC2)CCN(C)S1(=O)=O CC(C)C(O)CC(=O)NC(C)(C)CCC1CCN(C(C2(C)CC=CCC2)=O)CC1 c1(CC)nc2c(s1)C(N(C)C(=O)C(=O)NC1Cc3ccccc3NC1=O)CCC2 CN1C(=O)c2ccccc2C1CC(=O)NCCSC(C)(C)C C1(Cn2cc(C(CC)(C)O)nn2)C(C2CC2)CCN1C(=O)CCSC(F)(F)F NS(=O)(=O)c1cc(C(=O)NCC2(C(N3CCCC(F)C3)=O)CC2)c(O)cc1Cl c1(C(=O)NCC2CC(C)N(C(=O)CCC#N)C2)cccc2nccn12 N1(C(COc2c(C)cccc2)=O)CCC(CNC(C2C(C)C2C)=O)C12CCC2 C1(NC(=O)NC(C(C)C)C)COCCN(C(C)Cc2cccs2)C1 c1(C(C)C)[nH]ccc1C(=O)NCC1(F)CC(NC(=O)CCCc2ccccc2)C1 c1(CC)c(C(=O)NC2CCCN(C(=O)C=CC3CC3)C2C)cccc1F N=c1nc2cc(C(=O)Nc3cccc(NC(C45CC6CC4C5C6)=O)c3)ccn2[nH]1 C(N=c1cc(C)nc(-c2ccccn2)[nH]1)c1ccc(OC)c(C)c1 Cn1c(=O)sc2cc(C(N3CCC(CC4CCOC4)C3)C(=O)NC3CC3)ccc12 N1(C(c2cc(C3CCC3)no2)=O)CC(C2CCN(C(C3CC4CC3C4)=O)CC2)C1 C1(CC)CC2CCC(C1)N2C(=O)CC1CCCN(C(c2ccc(C)cn2)=O)CC1 N1(C(CCCCC#C)=O)CC(CNC(=O)C(=C2CCCCC2)F)C2CCCCC12 C(c1nc(C)c(C)[nH]1)=CC(=O)NCC1(NC(c2c[nH]c(=NC)s2)=O)CC1 C1(NC(c2cccc(CNC(c3[nH]cc(C)c3)=O)n2)=O)CCn2nnnc2C1 c1(C(=O)NCC(C)(C)NC(CCCc2n(C)cnn2)=O)cc(Cl)c(Cl)[nH]1 C12(NC(C3(SC)CN(C(C4(C)CCC(=O)CC4)=O)C3)=O)CCCN(CCC1)C2 CC(CC(=O)NC1CC(F)CN(C(=O)CCCc2cc(F)ccc2F)C1)C(F)F C(=O)(C1=CCCCC1)N1CC(COC)(CN(C(=O)CC2(C)CC(F)(F)C2)CC)C1 C=CC(O)C(C)(C)C(=O)N1CC2(CC(C(N3CCC(C(=O)O)C(C)C3)=O)CO2)C1 c1(C(N2CC(NC(C(CC)OC)=O)C3(C2)CC3)=O)ccc(CSC)c([N+](=O)[O-])c1 C(=O)(C1=CC2C=CC1C2)N1CCC(CC(NOCC(C)(C)O)=O)CC1 CCCCC(C(=O)NOCC(C)CC)NC(c1cn(C2CC2)cn1)=O C(=O)(C1=NOC(CNC(C2CC3(CCC3O)C2)=O)C1)NC(C(N)=O)CO c1(C(=O)NC(C(C)NC(=O)C(N)=O)CCc2ccccc2)cc2cccnn2n1 CCCCCCC(CC)(CC)C(=O)NC(C1CCNC1)CC C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CN(C(C2C(C)C2)=O)CC1N=[N+]=[N-] C1(NC(C(CC)N(CC)CC)=O)CN(C(=O)Cc2nonc2C)CC1C Cc1cc(F)ccc1C(F)(F)C(=O)NCCC(C)NC(c1cc(CF)on1)=O c1(CC(=O)NCCCCC2CCN(C(C3CCCCC3)=O)CC2)nc([N+](=O)[O-])n[nH]1 c1(C(N2C(CNC(C(N)=O)=O)C=CC2)=O)ccc2c(c1)OCC2 N1(C(C#CC(C)C)=O)CCC2(CCCCC2NC(c2ccoc2Cl)=O)C1 N1(C(c2c(CC)csc2)=O)CCCC1C1CCCN1C(c1cc(F)ccc1Cl)=O c1(C(=O)NCCN(C(c2ccc(CC)cc2)=O)C2CC2)c2c(nn1C)CCSC2 C(CNC(=O)C(=O)Nc1ncc[nH]1)(CC(C)C)NC(CC=CC=C)=O N1(C(c2[nH]c(CC)c(Cl)n2)=O)CC2CC1CCC2NC(C1(CCO)CC1)=O c1(NC(C)=O)sc(C)c(C)c1C(=O)NCCN(C(C1CCCS1(=O)=O)=O)C1CC1 C12(CNC(C3(C(=O)NC)CCC3)=O)CCCC1CN(C(=O)Cc1n[nH]cc1Cl)C2 n1(CC)cnc(C(=O)NC(C(=O)N(CCC(=O)NC(C)C)C)C2CC2)c1 CC1CN(C(=O)Cc2cn(C)nn2)CCC1Nc1cc(C(C)(C)C)ncn1 N1(C(CCCC)=O)CC(NC(c2nc(-c3ccccc3)oc2C)=O)C2(CCC2)C1 c1(CC)nc(C)c(C(N2CC(F)CC2CNC(=O)C(c2ccccc2)C)=O)o1 c1(C(=O)NCC(CO)NC(c2ccc(N)c(C)c2Cl)=O)cc2c(nn1)CCCC2 N1(C(C2(CC)CC2(F)F)=O)CCC(O)(C(C)NC(c2ccc([N+](=O)[O-])s2)=O)CC1 C1(CNC(C=CCCC)=O)CC2(CC2)CN1C(C1C2CC3C(C2=O)C13)=O N1(C(C2C(C)SCCC2)=O)CC2(CC(CC(=O)NCC3CCC(=O)NC3)C2)C1 N1(C(C2(CC=C)CCC2)=O)CC(C=C)(CC(=O)NC2(CO)CCC2)C1 Cc1ccccc1CN1CCN(C(=O)C(=O)NC(C2CC=CCC2)C)CC1 N1(C(C(C2CN(C(c3c[nH]c(=N)o3)=O)C2)OC)=O)CC(COC)C1(C)C c1(CC(=O)NCCC(C)NC(COC)=O)cc(F)cc([N+](=O)[O-])c1 C1(c2n(C)c(N3CCC(N4CCC(F)(F)CC4)CC3)nn2)CC2(CC(=O)C2)C1 c1(C(N(C)CC2CCCC(NC(COCCC=C)=O)C2)=O)csc(=NCC)[nH]1 c1(C(N2CCC3(NC(=O)C=CC4CC4)C(C2)C3)=O)cc2ccccc2[nH]1 C(=O)(C(F)C(C)C)N(C(CNC(c1ccn(CCCC)n1)=O)C)CC C1(CNC(c2c(C)cc(O)nc2)=O)CC2(CO1)CN(C(=O)C(C)S(N)(=O)=O)C2 C(=O)(C1=NOCC1)NC(C(C)NC(=O)CCc1ccccc1)(C)C c1(C(CC(=O)OCC(C(=O)OCC)O)c2cccs2)cc(C)nc(C)c1 C=CCCCC(C(=O)NCC(COC)OC)NC(c1ccc(C(F)F)o1)=O c1(C(N(C2CCCC2)CCNC(=O)CSC(F)F)=O)cccc(Br)c1Cl Cc1cc(C(N2CCOC(C(C)NC(=O)CNS(=O)(=O)C3CC3)C2)=O)cn1C N1(C(c2cc(C)cc(F)c2)=O)CCCC(NC(c2ccn(C)c(=O)c2)=O)C(F)C1 S(=O)(=O)(C1CCC(=O)CC1)N1CC(NC(c2c(I)ccc(C)c2)=O)CC(F)(F)C1 C12(NC(c3ns[nH]c3=O)=O)COCCC1CN(C(=O)COc1cccc(F)c1)C2 c1(C(N2CC(NC(C(C=C)C)=O)C3(C2)CC3)=O)cc(C)c(OC)c(C)c1 N1(C(=O)CCc2cn[nH]c2)CC2CC(C1)CN(C(c1ccc(O)nn1)=O)C2 C1(C)(CC)C=C(C(=O)NCC2(C)CCCN2C(=O)Cc2c(Cl)cnn2C)C1 Cc1nnc2n1CCC(C(N1CC(CNC(=O)CCc3cccnc3)C1)=O)C2 C1(NC(=O)CC2C=CCCC2)CCC(O)CN(C(=O)Cc2csc(C3CC3)n2)C1 C12(C(N3CCC(C)C(N(C(=O)C=Cc4ccsc4)C)C3)=O)CCC(CC1)C2(C)C c1(CC(N2CC(N3C(=O)CC(NC(C=CC)=O)C3)C2)=O)ccc(C)c([N+](=O)[O-])c1 C1(NC(CN(C2CC2)CC)=O)C(C)CN(C(C2(OC)CCC2)=O)CC1C C=C(C)C1OCCCC1C(=O)NCC12CCC(NC(=O)C(O)CC(C)C)(CC1)C2 C1(N(c2cnc(C)s2)C(C(c2ccccc2)OC)=O)CCCC12CCNCC2 N1(C(COCC)=O)CCC2(CCCN(C(=O)C(c3cnc(O)nc3O)(F)F)C2)C1 Cc1ccc(F)c2oc(C(=O)OCC3CC(C)(C)OC(C)(C)C3)cc12 C(=O)(C(C)(C)CC1CCOCC1)N1CC(O)(CNC(CC2C(C)OCC2)=O)C1 S(=O)(=O)(c1cccc(N2CCSC3(CCC3)C2)n1)NCC1CCCN(C)C1=O C(=O)(C(CCC1CCC1)NC(=O)C(C)C(F)F)NC(c1nc(=O)o[nH]1)C CCC(C(=O)N1CC(C)(CC(=O)N(C(C)C)Cc2cccnc2)C1)N(C)CC c12ccc3nc([nH]c3c1)CNC2=O.CC1(C)COCC(CC(=O)O)O1 c1(C(N2CCC(NC(C(C3CC(F)(F)C3)OC)=O)C2)=O)nn(C)c(N)c1C C=C(C)C(C)(O)C(=O)N1CC2(C1)CN(C(c1ccc(C(C)C)nc1C)=O)C2 N1(C(c2n(CC)ccn2)=O)CCCC(C)C1CNC(c1ccn(CC)c(=O)c1)=O Cc1nc(NCC2CC(C)(C)CCO2)cc(NC2CC2C2CCC2)n1 C(C(=O)N1CCCc2nncn21)C1OCCN(C(C(C)Cc2ccco2)=O)C1 N1(C(CSC)=O)CCN(C(=O)C(Cc2ccccc2)N(C)C(C)=O)C2CCC12 N1(C(c2ccc(C)s2)C(=O)NCC(C)C)CCOCC1C1CCCO1 c1(C(N2CCC(C(C)NC(Cn3c(C)ncc3)=O)CC2)=O)cc2cnn(C)c2s1 C(=O)(C1=COc2ccccc2O1)NC1CC(C)(NC(C(CCC)O)=O)C1 N1(C(=O)NC(C2CCOC2)C)CCn2c(nc3c2CCCCC3)C1 N1(C(c2c(C)ccc(F)c2)=O)CCC(NC(C2(F)CCOC2)=O)CC(C)(C)C1 c1(NCC#C)cccc(C(N2CC=CC(NC(C3(C(N)=O)CCCC3)=O)C2)=O)c1 N1(C(c2cnc(C)nc2)=O)CCOC2CN(C(=O)C(C)O)CC12 CC1(CNC(C2CNC(=O)C2)=O)CCCN1C(c1ccsc1-n1cnnn1)=O Cc1cccc(C(=O)NCC(N2CCN(C(C3(CC(C)C)CC3)=O)CC2)C)c1O N1(C(C(C=C=C)C)=O)CC(=O)NC2CN(C(=O)CCc3nc(C)cs3)CCC12 C1(CCNC(CCCNC(=O)OC)=O)(NC(c2csc(F)c2)=O)CCOCC1 N1(C(CCCN=[N+]=[N-])=O)CC(CO)C2(C1)CN(C(c1nc(=O)cc(N)[nH]1)=O)C2 Cc1cc(Br)ccc1NC(=O)C=C1CCN(Cc2cccc(I)c2)CC1 C1(C)(CNC(CC(COC)NC(C23CCCN2CCC3)=O)=O)CCCCCC1 c1(C(=O)NC(c2ccc(Br)c(Cl)c2)C)n[nH]c2ccc(C#N)cc12 CC1(C)COC(CC(=O)NCC2CCN(C(=O)CCc3cnoc3)CC2)C1 c1(C(=O)NCC2CC(NC(c3n(CC)ncn3)=O)C2(C)C)ccc(C#N)cc1C C1(CC)CCCCC1C(=O)NCCCC(C)NC(c1cnc(C(C)(C)C)nc1)=O c1(C(=O)NCC(CNC(c2cn(CC)nc2C)=O)(C)C)cccn2c(C)nnc12 c1(CC)cncc(C(N2CC(C(C(=O)NC(c3[nH]c(C)nc3C)C)OC)C2)=O)c1 N1(C(CN(CCC)C)=O)CCC(NC(=O)C(C)(C)C2CCCO2)C(CC)C1 C1(C(=O)OC)CCc2nc(C(=O)NCC3CC4(C3)CC(CSC)C4)ncc2C1 C=CCC(CC(C)C)C(=O)NCC(C)(C)CC(=O)NCc1nnnn1CC CCC(C)C(C(=O)N1CC2(CC(NC(=O)CNC(=O)C3CC3)C2)C1)NC(N)=O c1(C(N2CC(NC(Cn3c(C)cc(C)n3)=O)C3(C2)CC3)=O)ccc2c(c1)CCO2 c1(OC)ncccc1C(=O)NC(C)(C)C(=O)NCCN(C)C CCC(F)(F)C(C)(C)C(=O)NC1CCC1CNC(c1[nH]cc2c1CCS2(=O)=O)=O Cn1ncc(CCC(=O)N2CCC2CNC(=O)C(C2(O)CCCC2)F)n1 C1(NC(c2c(C)cco2)=O)C2CCC1CN(CC(F)(F)F)C2 C1(CC(N2CC(CC(C(=O)NCC(C#C)CC)F)C2)=O)CCCN(C)C1 c1(C(N2CCCC(NC(CCNC(C)=O)=O)CCC2)=O)nc2cc(F)ccc2s1 c1(C(=O)NC(CNC(C(C)n2ccnn2)=O)C(C)(C)C)ccc(F)c(F)c1O C1(CC(N2C3C(NC(c4c(C)nc(C)[nH]4)=O)CC(C3)C2)=O)CCC2(CCC2)CO1 O=S(=O)(c1ccc(NCC(O)CF)cc1Cl)NC1(c2ccc(F)cc2F)CC1 c1(C(=O)NCCCN(C(C(COC)(C)O)=O)C)csc2nnsc12 N1(c2c(S(C)(=O)=O)cccn2)CCC2(CCCCN(C(=O)CC(F)(F)F)C2)C1 c1(CC(=O)NC(C(C)NC(C23OCC(COC)(C2)C3)=O)CO)c(C)cccc1C Cc1cc(C)c(C(N2CCC(O)(CCNC(c3coc(Cl)n3)=O)CC2)=O)cn1 CC1CN2CCCCC2CN1C(=O)CCc1cccc(F)c1Cl c1(SC(C)C(N2CCCCC(NC(C3CC3F)=O)C2)=O)ccc(C#N)cc1 CCCCC(C(=O)N(CC(C)(C)CNC(=O)CC1C=NN(C)C1=O)C)C(C)C C1(CNC(C(C)=CCN)=O)CNC(=O)C1(C)C N#CC1CN(C(C2C3CCN(C(C4(NC5CC5)CCC4)=O)CC23)=O)CCO1 C(=O)(CCS(=O)(=O)N1CCOCC1)N1CC(NC(C(C=C=C)C)=O)C(O)C1 c1(C(=O)NC2CCC23CN(C(c2nn[nH]c2Cl)=O)C3)ccc2cc[nH]c2c1 CCCC(C1CC1)NC(=O)N(CCC)CC1CC1 CCC(CCOC)C(=O)NCC1C2CC1N(C(c1c(C(F)F)nn(C)c1C)=O)C2 c1(SCC(=O)NC(CNC(C(c2ccc(OC)cc2)C)=O)C)cc(C)ccc1C C=C=CCCC(=O)NC1CCC1NC(=O)C=CC=CC C1(N(C(C=CCOC)=O)CCOC)CCN(C(=O)CCc2cnoc2)CC1 N1(C(Cc2c(C)non2)=O)CC2CC1CC2NC(=O)CCc1ccc(Br)nc1 C(=O)(C1=CC2CCCCC12)N(CCCNC(CC(C(=C)C)OCC)=O)CC c1(C(N=c2[nH]n(C)c(Cl)c2)=O)cnc2n[nH]c(C3=COCCC3)c2c1 c1(CNC(C2N(C(C(CC)N(CC)CC)=O)CC2)=O)cncc(N)n1 c1(C(=O)NC23CC2CN(C(c2cnc(-c4ccco4)s2)=O)C3)cnc2sccn12 C(=O)(CCCC(CC)CC)N1CC(C(C(N2CCC(CC=C)C2)=O)OC)C1 C1(C(N2C(C(C)(C)C(=O)NC3CCOC3CC)CCC2)=O)CCCC2(CCC2)C1 C1(NC(C(C)=O)=O)CCCC1CNC(=O)C=C1CCCC1 c1(C(N2C3CC(NC(c4cc(C)[nH]n4)=O)C(C3)C2)=O)cc(F)cc2c1NCCC2 c1(C(N2C3(CNC(c4c(C(C)C)scn4)=O)CC(C2)C3)=O)cc(F)cc(N)c1F c1(C(=O)NCCCCNC(C(C)NC(=O)C(C)(C)C)=O)cnn(C)c1S(N)(=O)=O c1(C(=O)NC2C(NC(c3c(C)n(CC(C)C)nc3)=O)C2)cncn(C)c1=O c1(C(=O)NC2C(NC(C3(NC(N)=O)CC3)=O)CC2)ccc(-c2cnccn2)cn1 Brc1ccc2c(c1)C(NC1CCNCCC13CCC3)CCO2 N1(Cc2ncn(C)n2)CC(NC(c2cc(Cl)cc(Br)c2)=O)C(F)(F)C1 C(=O)(C1=NOC(CNC(=O)C=C(C)c2ccco2)C1)N(C1CCCC1)CC N1(Cc2c(CC)onc2C)CC2CC1CN2C(c1coc(C(C)C)n1)=O C(=O)(C1CCCc2nccn21)NCC1(C)CCCN(C(c2cnnc(O)c2)=O)C1 C1(N(c2nc(OC(=O)CC3CCC(C)CC3)sc2)C(C)=O)C=CS(=O)(=O)C1 Cc1ccc(C(N2CCCN(C(c3csc(C)c3N)=O)CC2)=O)cc1C CC(C)(C)CC(F)C(=O)N1CCC(C)(CNC(=O)C(O)Cn2cncn2)C1 CC1CC(C(N2CC(Cc3ccoc3)C2)=O)N1C(=O)CCc1ccsc1 S(=O)(=O)(c1[nH]c(=NC2CCN(C)C2)ccc1Br)NCC1C(C)CCNC1=O C#Cc1cc(C(=O)NC2C3CCN(C(=O)Cn4cncn4)CCC23)cc(F)c1 C(=O)(C(CNC(C1CC=C(C)CC1)=O)C(C)(C)C)NCCS(CC)(=O)=O C1(CC(=O)NCC(C(C)C)NC(c2cc(COC)on2)=O)CCC2CC2C1 CC1(C)CN(C(C2(CF)CC2)=O)CC1CNC(C1CCCNC1=O)=O CC(C)(CC(=O)N(CCO)CC1CC1)NC(=O)C(F)=CC1CC1 C1(OC)CCC(C(N2CC(F)(C(=O)NOCC(C)(C)O)C2)=O)C1 c1(CC(=O)NC2C(CNC(c3cnc(SC)s3)=O)CCC2)cnn(C)c1C C12(C(N3C4(C(=O)NCCC(C)CO)CC4CC3)=O)CCC(CC1)CC2 n1(CC(=O)NCC2CN(C(C(C)C)=O)C(C)(C)C2)nc2n(c1=O)CCCCC2 c1(OC)ccc(O)c(C(=O)NC2(C3CN(C(=O)C(O)C(F)F)C3)CC2)c1 N(C(=NCCF)N1CCC(CN2CCOCC2)C1)CC(N(CC)OC)=O CC(CN=C(NCC1C=CCC1)NC1CCCC1)Oc1ccc(Br)cc1 c1(C(=O)NCC(CNC(CCC)=O)CO)ccc(-n2ccnc2)c(F)c1 N1(C(CNC(CC)=O)=O)CC(C)(OCC(=O)NC(c2cnn(C)c2)C)C1 C=C(C)C(CC(=O)NCC1CCC(C(=O)NC(c2cncnc2)C)CC1)OCC N1(C(CCCCOC)=O)CCCC(C)(CNC(c2c(OC)cccc2F)=O)C1 N1(CC(=O)N(C)CCc2ccccc2)CCOC(CO)C1 c1(C(N2CC(NC(C=CC(CC)=CC)=O)CC2(C)C)=O)cc(S(N)(=O)=O)oc1Cl N1(C(CCOC(C)C)=O)CCC(CO)C(NC(c2nn(C(F)F)cc2Cl)=O)C1 C1(NC(c2ccc(NC(C)=O)o2)=O)CCCC(CNC(C2CC3(CSC3)C2)=O)C1 c1(C(=O)NCCC(N2C(CNC(CC(CC)C)=O)C=CC2)=O)cc(C)ccc1C N1(C(C(CC(C)C)ONC(c2c(OC)cncc2)=O)=O)C2CCC1CC(=O)NC2 CC(CC1=CCCCC1)N(c1nnc(-c2cnccn2)n1CCC#N)C c1(C(=O)NC2(CF)CCN(C(C(C(C)C)(C)O)=O)C2)ccc(P(C)(C)=O)nc1 C(=O)(C(C)C(O)CCCC)N1CCC(C(N2CC(C#C)C(OC)C2)=O)(CF)C1 c1(C(N2CCCC(CCNC(C(COCC)(C)C)=O)C2)=O)cnc(Cl)cc1N N1(C(=O)CCOCC2CC2)CC2(CCN2C(=O)Cc2ccnn2C2CCCC2)C1 c1(C(C(=O)NCC(=C)C)N(C2CC2)C2CC2)cccc(F)n1 O=C(C(O)C1=CCCCC1)NC1(C(N2CC3CCC2C3)=O)CCSC1 N1(C(C(CC)N(C)C(C)=O)=O)CCC(C)N(C(=O)COc2ccc(F)cc2)CC1 C1(COC)(NC(c2ccc(OC)nn2)=O)CCN(C(=O)CC2CC3(CC3)CO2)C1 N1(C(Cn2c(C)cc(C)n2)=O)CCN(C)CC1CNC(=O)C#CC(C)(C)O CC1CN(C(c2cc(O)ccc2Br)=O)CCN1C(c1ccc(C2CC2)s1)=O c1(C(=O)NC(CNC(COC)=O)(C)C2CCC2)csc(C(F)F)c1 Cc1c(C(=O)NC2(C)CCN(C(C3COC(=O)O3)=O)CC2)oc2ccc(Cl)cc12 N1(C(c2c(C)noc2)=O)CC2CCC1CN2C(=O)C(C)CC1CC1 C1(OC)CC2(C1)CN(C(=O)C(C1CCCO1)NC(=O)C(n1ccnc1C)C)C2 c1(CC(C(=O)N2CC(CNC(C(C)OCC#C)=O)C2)C)ccc(OC)cc1 N1(C(c2cnc(SC)s2)=O)CCOCC1CN(C(=O)CC1(C)CC1)C Cc1cccc(N)c1C(=O)NC1CCN(C(c2cnn(C3CCC3)n2)=O)C(C)C1 C1(NC(C=Cc2n(C)ncc2)=O)COC2(CCCN(C(c3cccs3)=O)C2)C1 C1(N(C(C(c2ccccc2)SC)=O)C)CC2CCC(C1)N2C(=O)C1=CCCO1 CCC(C#N)C(=O)N1CC(N(C)C(c2nn(C)cc2C)=O)C1 Cc1cc(F)c(NC(C2CC(C)(C)CN2C(=O)CCCN2CCCC2)=O)cc1C N1(C(C2CC(OCC)C2)=O)CCCN(CCNC(c2cocc2C(N)=O)=O)CC1 c1(C(N(CCNC(c2c(C)csc2)=O)C2CC2)=O)cc(N)ccc1Br N1(C(C(CC(C)C)ONC(C(C)=CCC)=O)=O)CCc2c(C#N)cccc21 Cc1nnccc1C(N1CCCCC1CCNC(=O)CC1CN(C)C1)=O c12ccc(cc1)N(C)C2C(=O)NCc1ccc(C)s1.N1(CC(=C)C)CCCC1 n1(CC(=C)C)nnnc1C(c1sccc1Br)NCC1CCCOC1 c1(N(C(c2c(C(C)C)scn2)=O)C)cc(-n2ccnc2)ncn1.C12CCCN1C2 c1(C(=O)NC2CC(NC(c3cc(OCC)n[nH]3)=O)C2)ccc2cnnn2c1 C12CCCCC1CC(=O)N2.C1(NC(=O)OC(C)(C)C)(CNC(C2CC2F)=O)CCC1 N1(CCOC)CCN(C(=O)C(=O)NCc2nc(C)cs2)CC1 c1(C(=O)NCC2(COC)CCN(C(C(CC)F)=O)CC2)cn2ccccc2n1 C1(CNC(c2ccc[nH]2)=O)COCCN(C(=O)CC2C=CCC2)C1 c1(CC(=O)NCC(C)(CO)NC(COCCC)=O)cccc(Cl)c1O.SCC C(=O)(CC(C)(O)COC)N1CCCC(C(N(CCOCC)CC)=O)C1 CCCC(C#N)C(=O)N1CCCC(CNC(=O)CCn2ccccc2=O)CC1 C1(CC(N2CC(CN(C)C(c3cc[nH]c3C3CC3)=O)C2)=O)CC2(CCC2)CO1 C1(C(N(C(c2cc(C)on2)C)C)=O)CC12CCN(C(c1cc[nH]c1C)=O)C2 C1(C(N2CCC(C(C)C(=O)N(CCO)CCO)CC2)=O)CCC=CCCC1 Cc1ccc(OC(C)C(=O)NCC2CC(F)(F)CN2C(=O)CC(C)(C)O)c(C)c1 C1(c2ccc(CC)o2)CN(Cc2ccc(OCC#N)cc2)CCO1 C=C(C)CCCC(=O)N1CCCCCC1CNC(=O)C(c1c(C)cccc1C)O N1(C(C=C(C)C(F)F)=O)CCOC(CN(C(=O)CC2CCC3CC23)C)C1 N#CC1CN(Cc2nc[nH]c2C(C)(C)C)CCN1C(c1cccc(Cl)c1F)=O C(c1ccc(Cl)c(Cl)c1)=CC(N1CC(CC(=O)N(C)Cc2cccnc2Cl)C1)=O Cc1cnn(C)c1C(=O)NCCc1cc(C(=O)NCCCCCCO)no1 Cc1c(C(=O)N(CCC#N)CCc2nn[nH]n2)oc2c(F)cccc12 C1(F)(C(=O)NCCc2c(Br)ccc(C)c2)CC2CCC(C1)N2C(=O)OC(C)(C)C C(=O)(C(O)CCS(C)=O)NC1C2CN(C(CCCOc3cccc(C)c3)=O)C1C2 C1(C(=O)NC2C(C#C)N(C(=O)OC(C)(C)C)CC2)CCn2ncnc2C1 c1(C(=O)NC(C)CCNC(C2(N(C)C)CCCCC2)=O)cc(O)cc(Br)c1 C(=O)(C1COc2ccccc21)NCCCNC(C1C(NC(=O)OC(C)(C)C)C1)=O C1=CC(=O)NONS(=O)C(=O)N2C1CCC2.C1(=CC#N)CC1(F)Cl N1(C(CN(C(=O)OC)C)=O)CCCN(C(c2nccnc2N)=O)CCC1 C=CC(C)CC(=O)NC(CCSC)C(=O)NCC1CC(C)(C)C1 c1(N2C3CN(C(c4cc(C)nc(C)n4)=O)C(CC3)C2)nccc(C)c1[N+](=O)[O-] C1(N(C)C(c2cnn(CCNC(=O)Cn3ncnn3)c2)=O)CCOCC1F C(C(C(=O)NCC(=O)OC)C(C)(C)C)NC(CC(C(C)C)OCC)=O c1(NC(c2csc(Cl)n2)=O)cccc2c1CN(C1CC1)C2=O C#Cc1ccc(C(=O)NCC2C(C)CCN2C(=O)CNS(=O)(=O)C2CC2)c(F)c1 n1(CC(=O)N(CC2CCN(C(C3C(COC)C3)=O)CC2)CC)cc(S(N)(=O)=O)cn1 c1(C(=O)NC2C(C)(C)CN(C(C3CCC(=O)N3)=O)C2)csc(S(N)(=O)=O)c1 C(=O)(CCCC(F)(F)F)N(CC(=O)NCC1CCC=CCCC1)CC Cc1ccsc1C=CC(=O)NCC1CCC1NC(=O)C(C)C1CC1 C1(C(=O)OC)CC(C)N(C(=O)C(C2CCC(C)(C)CC2)CN)CC1C C1(C2CCN(C(c3coc(O)n3)=O)C2)(NC(CC2N(C)C(=O)CC2)=O)CC1 c1(C(N(CCN(C(C(C)OCC)=O)C)C)=O)sc(C2CCCCC2)nc1C c1(OC)cc(C(N2CCC(NC(c3cnc(Cl)cc3Cl)=O)C(O)C2)=O)ccc1Br N1(C(CNC(c2c(C)occ2)=O)=O)CCN(C(=O)CC2(C)CCCC2)C2(CC2)C1 CCCCCCC(C)C(=O)N1CCC(CC(=O)NC(CN(C)C)C(C)C)C1(C)C C(=O)(CCCC(C)(C)CC)NCC(CNC(c1n(CC)cnn1)=O)C CC1CN(C(=O)C(C)(C)C#N)CCN1C(=O)C=Cc1cncc(F)c1 CC1(C)CC(CNC(C2(C)CCCS2)=O)CN1C(=O)Cc1cccnc1 C1(CC)C(NC(c2coc(C)c2)=O)CCCN1C(=O)C(C)N1CC(C)C1 CCCCCC(C)CC(=O)N1C2CCC1CN(C(=O)Cn1nnc(=N)[nH]1)C2 c1(C(=O)NC(CC(C)NC(c2cncc(C)c2)=O)C)cc(N)nc(Cl)c1 CCC(CC(F)(F)F)C(=O)NC(CNC(=O)CC1CCC1)C1CCC1 C=C1c2ccccc2C(=O)N1CCC(=O)NCC1OCCC12CCNCC2 Cc1c[nH]c2ccc(OS(=O)(=O)CC(C)Oc3ccc(Br)cc3)cc12 c1(C(C)Nc2c(C)ccc(OC)c2)oc2ccccc2c1C C1(NC(C2C(CC)CN(C(C3CCS(=O)CC3)=O)C2)=O)CCOC12CCCC2 C12(CCNC(CC3(C=C)CC3)=O)CCC1CN(C(C1(C)CS(=O)(=O)C1)=O)C2 c1(-c2cn(CCN(C(=O)CC3CCC(C(F)(F)F)O3)C)nn2)cccc(C#N)c1 C1(=O)C(N(C)C)CN1.C(C(=O)N(C(C)C)CC)OC(C1(OC)CC1)=O c1(C(N(C(C)CCNC(=O)CC2CCNC2=O)C)=O)c[nH]c(=O)c2ccnn12 C1(CC)CN(C(C2(COC)CCC(=O)N2)=O)CCN1C(c1cccc(SC)c1)=O c1(C(N2CC3C(NC(C4CCC(=O)C4)=O)(C3)C2)=O)cc2nc(Cl)ccc2s1 N1(C(=O)OC)CCC(C(=O)NCc2cn(Cc3cnn[nH]3)nn2)C1C(C)C C1(NC(C(C(C)C)SC)=O)CC2(C1)CN(C(c1occc1C(C)C)=O)C2 Cc1cc(C(=O)NC2(C)CC(NC(=O)C(C3CCC(=O)N3)C)C2)co1 FC1(F)C2CCC3C(C2)C13CN1CCSC12CC(C(F)F)C2 c1(C(=O)NC2C(C)CCN(C(C(CNC(C)=O)(C)C)=O)C2)cc(S(N)(=O)=O)co1 Cc1cc2ccc(C(=O)NCCC3CCCN3C(C3CCCCCC3)=O)cc2o1 C1(CC(N2CC(CCNC(c3c(CC)ncs3)=O)(OC)C2)=O)CCCC2CC12 C1(CNC(C2C(C)C2)=O)CCCCN(C(=O)C(C)(C)COC2CCCC2)C1 n1(CC)nnc(C(=O)NC2(CNC(C3(COC)CC=CC3)=O)CCCCC2)c1C C(=O)(CCCC(C)NC(=O)C(c1cccnc1)N(C)C)NC(C)C(C)(C)CN(C)C c1(C(=O)NCCC(C)NC(C2C3(CC(OCC)C3)C2)=O)c[nH]c2c(C)cccc12 N1(C(Cc2nc(=N)[nH][nH]2)=O)CCC2(NC(c3ccc4nsnc4c3)=O)CCCC12 C1(NCc2n(Cc3sccc3)nnn2)CC2CCCC2C1 CCC(C#N)C(=O)NC1CCCC1NC(c1cc(C(N)=O)cs1)=O Cc1ccc(C(C)(CNC(=O)N(C2CC(O)C2)C)CO)cc1 C1(NC(C(C)C(C)O)=O)COC2(C1)CN(C(c1ccc(O)c(F)c1F)=O)C2 c1(CC(=O)NCC2C(NC(CCC(=C)C)=O)CC2)ccc2nc(O)[nH]c2c1 c1(C(N2CC(C)(NC(C=Cc3c(C)nccc3)=O)C2)=O)cc(F)c(C)c(N)c1F N1(C(c2nc(C)nc(O)c2)=O)CCC2(CC1)OCCC2NC(C1CCC1(C)C)=O C1(C(=O)NCC(C)O)(N(CCC(C)(C)C)CCO)CCCC(c2ccccc2)CC1 C1(NC(=O)C(=O)NC2CCN(c3ccccc3)CC2)CCNC2(CC2)C1 CC1CCC(CC(=O)NCc2cc(C(=O)NCc3nccs3)cs2)O1 C1(NC(Cn2nc(C)c(Cl)c2)=O)CC2CCC1N2C(c1snnc1C)=O N1(C(c2c(C(C)C)ocn2)=O)CCCCC1CNC(=O)Cn1cc(C2CC2)cn1 c1(CN(C(=O)C=C2CCN(C3CC3)CC2)C)ccc(F)cc1C(=O)O N1(C(C2(C#C)CCN(C(=O)C(C)C)C2)=O)CC2(CNC(=O)OC2)C1 C1(NC(=O)CCn2cnnn2)CC2CC1N(C(C1(COCCO)CC1)=O)C2 C1(CC)C(C(=O)NCC2(CCO)CC2)CCN1C(c1c[nH]c(C#N)c1)=O C(C(C(=O)NCC(O)CC(=O)OC)C(C)(C)C)NC(c1cc(COC)on1)=O C1(NC(C(CSC)OC)=O)CC(CNC(C2(F)CCOCC2)=O)C(O)C1 c1(C(=O)NC(CNC(C(CC#C)C)=O)(C)C2CCC2)cnc(O)c2cnccc12 CC(CC(=O)NC1CCC12CN(C(c1ccc(Br)o1)=O)C2)C(F)(F)F CC1CCN(C(c2cnc(N)c(Cl)c2)=O)CC1CNC(C1CN(C2CCC2)C1)=O N1(Cc2cc(OC)ns2)CC(NC(c2occc2Br)=O)CCC1C N1(C(C2CC(OC)C(OC)C2)=O)CCC(F)(CNC(=O)C(F)C(F)(F)F)CC1 Cc1n[nH]c2cnc(C(=O)NC3CN(C(c4ccc(Cl)cn4)=O)CCC3F)cc12 c1(-c2nc(CC(CC)C)nn2CCOCC(F)(F)F)ccc(Cl)c2occc12 c1(C(=O)NC2CCN(C(CCCCOC)=O)CC2F)cc(C)c(C)nc1C C1(CN(C(=O)CC2CC2C)CC)CCN(C(c2cc(C3(C)CC3)on2)=O)CC1 C1(C(=O)Nc2c(C)cccc2)CN(C(=O)C=CCF)CC12CC2 c1(C(=O)NC2(CNC(C(C)n3cccn3)=O)CCOC2)cc(Cl)ccc1N C1(CCNC(C(C=C)(C)O)=O)CN(C(c2cnc(C)cc2Cl)=O)CCS1(=O)=O Cc1nc(NCC2CC(C)N(C(C3OC(C)CC3C)=O)C2)c2ccsc2n1 c1(C(N(C2CCCN(C(C3CCN(C)C3=O)=O)CC2)CC)=O)nccc(Cl)c1F C(=O)(CC(CC)C(C)(C)C)N1CC(C)(NC(C(=Cc2ccc(F)cc2)C)=O)C1 c1(NCCC2CCN(C(C3(C)CC3)=O)CC2)nc2c(cc1C#N)CCC2 C1(NC(=O)CN2CC3CCC2C3)(CO)CCCN(Cc2ccn(C3CC3)n2)C1 c1(C(N2CCC(F)(C(=O)OCC(c3cc(C)sn3)=O)C2)=O)c(F)cc(F)c(F)c1F C1(N(CCC)C(C23CCC2C3)=O)CCN(C(=O)CSc2nncs2)CC1 Brc1ccc2c(c1)CN(Cc1cnc3[nH]ccc3c1)CC2 C(C)(CCCNC(c1cc(-c2ccco2)[nH]n1)=O)NC(C(c1cncnc1)C)=O c1(NC(C(C2CC(C)OC2)N2CCC(CN(C)C)C2)=O)ccccc1Cl c1(C(=O)NCC2CCN(C(C(C)(C)OC)=O)C2)c(Cl)cccc1Cl c1(C(N2CCC3(C(C(N(CCN(C)C)C)=O)C3)C2)=O)ccc(F)cc1C#N C1(NC(CC2N(C)C(=O)CC2)=O)CC2CCC1(NC(=O)COC1CCOC1)C2 C1(NC(=O)CN(C(=O)C(F)F)C2CC2)CCOCC1O c1(C(N2CCN(C(CC3C(CC)C3)=O)CC2CF)=O)cc(N)c(Cl)c(O)c1 Cc1cc(C(=O)NC2CN(C(=O)Cc3cncc(O)c3)CC2C)n2ncnc2n1 C1(NC(=O)Cc2noc3ccccc23)CN(C(=O)CC(F)F)C2(CCCCC2)C1 C(=O)(C(C(CC)=Cc1ccsc1)N(C)Cc1nncn1C)NCC=C c1(C(=O)NC(C2CCCC2)CNC(C(CSC)OC)=O)cc(Cl)ccc1C Cc1cc(Cl)cc(Cl)c1OCC(N1CC2CC(NC(=O)C=C(Cl)Cl)CC2C1)=O c1(C(C(N2CC(N(CC(=O)N(C(C)C3CC3)C)C)C2)=O)O)cnn(C)c1 C1(N(C(C(C2CCCOC2)OC)=O)CC(C)C)CCN(C(=O)C(C)(C)CO)CC1 c1(NCCC(=O)NC(C)C)ccc(S(=O)(=O)NC2CCN(CC(F)F)C2)c(Cl)c1 C1(c2nnnn2C)(NCc2cc(C)n(C)n2)C=CCC(C(C)(C)C)CC1 N1(CCCC(c2n(C)[nH]c(=N)c2)=O)CC(c2cnn(C)c2)C2(CCOCC2)C1 c1(C(=O)NCC2N(C(COC(CC)CC)=O)CCC(C)C2)nnn2c1CCCC2 C#CCC(C)(C)C(=O)N1CCC(C)C(CNC(C2(CC(C)C)COC2)=O)C1 CC1C(CNC(=O)Cc2ccc3c(c2)CC3)CCCN1C(=O)C(C)c1cccs1 CC1=C(C(=O)N2CCC(F)C(NC(=O)CC3CC(C)(C)CO3)C2)CCCO1 c1(C(N(CCNC(C(C)(C2CCC2)OC)=O)C)=O)nccc2occc12 N1(C(C2(OC)CCSCC2)=O)CCC(NC(=O)C=Cc2ncc(C)[nH]2)C(CO)C1 C1(NC(c2cc(O)ncn2)=O)CCC2(CC1)CC2NC(c1csnc1Cl)=O c1(C(=O)NCCC2N(C(C3C(C)C3)=O)CC(F)(F)C2)cn(C)cc(Br)c1=O C1(NC(c2n(C=C)nnc2)=O)CN(C(c2sccc2Cl)=O)CC1C1CC1 c1(C(=O)NCC2C(NC(C3(O)C(C)(C)C3)=O)CC2)ccc(S(=O)(=O)N2CCCC2)o1 CS(=O)(=O)C1CCC(C(=O)Nc2ccncc2)CC1.c12ccccc1[nH]c(=O)[nH]2 C1(NC(C(CC)(C)OC)=O)CCC2(CC1)CC(NC(=O)C=Cc1cn(C)nn1)C2 c1(C(=O)NC(C(C)C)(C)CNC(=O)C=Cc2ccnn2C)cccc2ncoc12 N1(C(c2nc(C)sc2C)=O)CCC2CC(CNC(=O)CNC=O)CCC2C1 CC1(C(=O)NCC2(C(N)=O)CN(C(c3ccnc(Cl)c3N)=O)C2)CCCCCC1 c1(C(=O)NCC(C)N(C(c2ccc(C)cn2)=O)CC)cc(OC)cc(C)c1 N1(CC(=O)NCc2cc(C)n(C)n2)CC2CN(C(=O)C(C(C)C)NC=O)CC12 N1(C(C2=CC(C)(C)C2)=O)CCCC(C2(NC(C3CCCC34CCC4)=O)CC2)C1 c1(C(=O)NC2(CCNC(C3(CC)CC3(F)F)=O)CCCC2)ccc2sccc2c1 n1(CCCC(=O)NC2CC(CCNC(C(C)NC(CC)=O)=O)C2)cnc(C#N)n1 C1(C2CN(C(=O)CCc3cn(C)nn3)C2)(NC(CC2N(C)CCC2)=O)CC1 c1(C(C(=O)NCC2(F)CC(NC(c3cc(C)n(C)n3)=O)C2)O)ccc(Cl)c(F)c1 C(=O)(NNc1oc(CC(C)C)nc1C#N)N1C(CC)CCC(C)C1 c1(C(=O)NCC(CNC(CNC(CNC(C)=O)=O)=O)CO)ncc(F)cc1F c1(CCC(=O)N(C2CC(C(=O)OC(C)(C)C)C2)C)ccc(CO)cc1 N1(C(C(P(C)(C)=O)O)=O)CCC2(CCC2)C(CNC(=O)CC2(O)CCCC2)C1 C12(CNC(C3CCS(=O)CC3)=O)CCCC1N(C(c1ccccc1F)=O)CCC2 N1(C(CC2N(C(C3C(C(C)C)CCO3)=O)CC2)=O)CCC(N(C)C)(CO)C1 C#CCC(CC(=O)N1CC(C)(C)CC1CO)NC(=O)C=CCO C(CCCCCNC(C1CC12CC(NC(C1CCOC1(C)C)=O)C2)=O)OC C(C1CCCN1C)=CC(=O)NCCN(C(c1nc(Cl)cs1)=O)CC CCCCS(=O)(=O)NCC(=O)N(C)CCN(C)C(c1cn(CCC)nn1)=O c1(COC)ccc(N)c(C(=O)NCC(C2CC2)NC(C2(C(C)(F)F)CCC2)=O)c1 CC(N=[N+]=[N-])C(=O)NC1CCCC(CNC(C2CCC(CCO)CC2)=O)C1 C1(NC(Cn2c(CCC)ncc2)=O)(CC)CCN(C(c2cc(CC)no2)=O)CC1 O=Cc1sc(CNc2cnc(F)cc2C(=O)NC(CO)C(F)(F)F)c(Br)c1Br C=CC1(C(=O)NCCC(=C)C)CCN(C(=O)C(C)S(N)(=O)=O)C1 C(=O)(C1=CCS(=O)(=O)C1)N1CCCC(NC(c2ncn(C)n2)=O)CC1 c1(C(N2C(C)CC(NC(C3(c4ccc(F)cn4)CC3)=O)C2)=O)ccc(N)c(F)c1 N1(C(CN2CCN(CC)CC2)=O)CC(C)N(C(=O)CNC(=O)NC2CC2)CC1C C(=O)(CC(C)CC(C)C)NCC1N(C(c2cccc(CC)c2)=O)CC(O)C1 CC1(C)C(CNC(C2CCO2)=O)CCN1C(=O)CSCCC(F)(F)F CC1(NC(c2cccn(O)c2=O)=O)CCCN(C(=O)CCn2ccnn2)C1 C(CC(C)C)(C(=O)NC(CNC(=O)C=CC(C)(C)C)CC(C)C)NC(C)=O N1(C(CC(CC)(C)C)=O)CCCN(C(c2coc(-c3ccccc3)n2)=O)C(C)C1 N1(CC)CCc2c(sc3nc(SCC(O)CN(C)C)nc(O)c23)C1 c1(C(C(=O)NCCCN(C(C(C)(C)SC)=O)CCO)F)cccc(C)c1 Cc1ccc(Cl)c(C(=O)NC23CC(CNC(=O)C4=COCCC4)(C2)C3)c1 C(=O)(C1CCCc2ccccc21)NCCC(C)NC(c1cc(CC(C)C)on1)=O Cc1ccc(OCCCC(=O)NC(C)CC(C)NC(=O)Cn2cncn2)c(C)c1 CC1(C)C(CNC(=O)CN2CCN(C(c3ccc(O)cn3)=O)CC2)C1(C)C N1(C(C=C2CCN(C)CC2)=O)CCC(C(F)(F)F)C(CNC(=O)C2=COCC2)C1 c1(C(CNC(=O)CCC2CC(C)CS2)OC)ccccc1C(F)(F)F C1(CC=C)(NC(c2ccc(C)c(C)n2)=O)CCCN(C(=O)C(N)=O)C1 N1(C(c2ccc(O)cc2OC(F)(F)F)=O)CCOC2CN(Cc3cscn3)CC12 c1(C(C(=O)N(CC(O)CNC(=O)CCc2ccccc2)C)OC)ccccc1Cl C#Cc1c[nH]nc1C(=O)NCC=CCC(=O)NCCC(C)C=C Cn1ncc(C(=O)NCC(=O)NCC2CSCCN2C(=O)CCCC#N)c1C c1(CC)cc(C)[nH]c(=NCC2CCC(NC(=O)C(C)S(N)(=O)=O)CC2)n1 C1(C(N(C2CCN(C(=O)CC3CCC(C)CC3)C2)CC)=O)CC(=O)NC(=O)N1 N1(C(C(C)N(CC)CC)=O)CCC(C(=O)NCC#CC#CCO)C12CC2 c1(COC)ccc(C(=O)N(CC(=O)NC(c2nnc(C)o2)C)C)o1 N1(C(C(CC=C)N(C)C)=O)CC(NC(=O)CCCC(OC)OC)CC1(CC)CC c1(C(C)C)cccc(NC(C2CC(NC(=O)CN3C(=O)CSC3=S)C2)=O)c1 CCC(F)(F)C(=O)NCCCN(C(=O)CC(n1nc(C)cc1C)C)C N1(C(c2cccc(CC)c2)=O)CC(F)(F)CC1C(=O)N(CC(C)(C)CO)C c1(NC2(c3n(CC)nnn3)CC(Br)C2)ccc(C(c2ccccc2)C(N)=O)cc1 CCCC(CCCNC(=O)CC1(O)CCCCC1)NC(=O)C(CCSC)OCC C=CC(C)(C)CCNC(=O)N(C)Cc1ccncc1C C(c1cnc(O)nc1O)=CC(N1CCCC(N(C(c2cnc(Cl)s2)=O)CC)C1)=O CC1(C(=O)NC2CCC(CNC(=O)CC(F)(F)F)CC2)CCC12CCC2 C(CO)(C(=O)NCc1cc(C(=O)NC2(c3nc[nH]n3)CCC2)cs1)OC C(=O)(C(F)CC(C(=O)OC)NS(=O)(=O)c1ccc(OCF)cc1)OC c1(C(=O)OC)ccc(C#CC(=O)C(c2cccnc2)C2CCCC2)cc1 C1(C(=O)NCC2CCC(=O)N2)CN(C(=O)CCc2cn[nH]c2)CC12CCC2 c1(CN2CC(CC(=O)Nc3cc(C(F)(F)F)no3)C2)ccccc1Br C(=O)(C1=COc2ccccc2O1)N1CC(CNC(c2cn(C)[nH]c2=N)=O)OCC1 N1(C(C(COCC)C)=O)CCCCCC1CNC(=O)CC(F)F c1(C(=O)NC2C(NC(C(C)OCCOCC)=O)C2)c(N)ccc(F)c1C C1(CNC(COCC(=C)C)=O)CC(C(=O)NCc2ncn(C(C)C)n2)CO1 n1(CC)nnc(C(=O)NC2(COC)CCN(C(c3conc3C(C)C)=O)C2)c1C C(=O)(C1CCCc2nccn21)NC1CCN(C(c2ccc(C#N)o2)=O)CC1CO C(=O)(CS(=O)(=O)c1ccccc1Cl)N(C(=O)CC1CCCC(F)C1)CC(F)F Cc1oc(C#N)cc1C(N1CCC(CNC(=O)C(C2CCC(=O)N2)C)C12CC2)=O c1(CC(=O)NC2(CNC(=O)C=Cc3ncc[nH]3)CCCC2)ccc(Cl)cc1 C1(NC(c2ccnc(C)c2C)=O)CN(C(=O)CC2CCC2)CC(F)(F)C1 C(=O)(CCCN(C)C(c1cscc1OC)=O)N(C(C)CO)CC C(=O)(C(C(C)(C)C)NC(C1CC=CCC1C)=O)N1CCC(CC(=O)NC)C1 Cc1nc2c(CC(=O)OC3CCCCCCC3)cccc2o1 CC1CN=C2NC(C(=O)N3CC4(C3)CN(C(c3ccc(Br)o3)=O)C4)=NN2C1 n1(CC(N)=O)ccc(=NC(=O)C(=O)NC2CCN(C(C3CCC3)=O)C2)[nH]1 C1(C(=O)NCCC2OCCC2C)(NC(CC2(CC)CCC2)=O)CC(F)C1 C1(C(C(N2CCC(Cn3c(C)ncc3)C2)=O)N2CCCC2)CC2CCC1O2 c1(C(N2CCC3(NC(c4cccnc4)=O)C(CC2)C3)=O)[nH]nc2ncnc(O)c12 C1(NC(CCCSC)=O)CC(C2CCN(C(c3cc(C)nc4ccnn34)=O)C2)C1 N1(C(C(c2ccc(N)cn2)C)=O)CC2(C)CN(C(C3CC(O)C3)=O)CC2(C)C1 C1(NC(c2ccnc(C(F)F)c2)=O)CN(C(C2(C3CCCO3)CC2)=O)CC1O N1(C(c2scc(OC)c2)=O)CC2(CCC(CNC(C3CCC(C)C3)=O)O2)C1 C1(=CC(=O)NCC(CC)NC(C2CCOCC2OC)=O)CN2CCC1CC2 c1(C(N2CC(O)(C(C)NC(c3cn(C)cn3)=O)C2)=O)ccc(Cl)c(C#N)n1 C(=O)(C1Cc2ccc(Cl)cc21)NC(C1CCCN(Cc2nccc(C)n2)C1)C CC1CC2(CCO1)CC2C(=O)NCC1C2CN(C(=O)CCCc3nccs3)CC12 c1(C(=O)NC2CC(NC(C=Cc3n(CC)ccn3)=O)C2)ccc2nnn(C)c2c1 CC1CCC1N=c1[nH]c2ccc(S(=O)(=O)N(CC(C)(C)CO)C)cc2s1 c1(C(=O)NC2CN(c3nc(C)cc(OC)n3)CC(F)C2)c(F)cc(C#N)cc1F c1(C(N2C(C)CC(NC(c3c(NCC)scn3)=O)C2)=O)cc(C)cc(Cl)n1 C1(C2CCC2)(C(N(CCN(C(c2n[nH]c(C)c2Br)=O)C)C)=O)CC1(F)F Cn1ccc(-n2cnc(C(=O)NCCNC(=O)CCN(c3ccncc3)C)c2)n1 Cc1cc(C)n2ncc(C(=O)NCCC(C)N(C)C(C3COC3)=O)c2n1 C1(NC(C(C)(C)n2cc(Cl)cn2)=O)COCCN(C(C2COCCC2(F)F)=O)C1 c1(C(c2ccccn2)N(C(=O)CNC(=O)Cn2cccc2)C)ccc(F)cc1 C1(NC(CNS(NC)(=O)=O)=O)CC2CC1N(C(=O)C(C)(CO)NC(C)=O)C2 N1(C(CC(CC)SC)=O)CC(C2CN(C(=O)C(CC)CCOC)C2)C1 CC1CNc2c(C(=O)NC3CCCCC3CNC(c3csnn3)=O)cnn2C1 C1(C(=O)NCC(C)SC)Cc2ccccc2O1.c12nc(cc(O)n1)NC2=O N1(C(C(CC)(C)F)=O)CCCCC2(CCN(C(c3cc[nH]c3C)=O)C2)C1 N#Cc1ccc(OCC(=O)NC2CC(NC(C3CCC=CCCC3)=O)C2)c(Cl)c1 Cc1nc2ncnn2cc1C(=O)NC1CC(O)CN(C(=O)CC2CC=CCC2)C1 C(=O)(CCCC(=O)NC1CCCN(C(c2n[nH]cc2Br)=O)C1C)NCC c1(OC(C)C)cc(C(=O)NC2CC(N(C)C)C2)ccc1F.C12CCCN1C2=O C(=O)(N=c1cc2n([nH]1)CCCC2)C1C(CC)N(C(C23C(=O)C4CC2C3C4)=O)CC1 c1(C(N2CC(OCCNC(C(CC)F)=O)C2)=O)n[nH]c2c1COc1ccccc1-2 n1(CCC)ncc(C(=O)NCCN(C)C(C2(CO)CC2(F)F)=O)c1Cl C1(CNC(C(CC)F)=O)CN(C(c2[nH]cnc2C)=O)CC(C)(C)O1 c1(SN2CC=C(C)C2)nc(C)cc(=NC(C)c2ccc(-c3cc(F)cc(F)c3)cc2)[nH]1 N1(C(c2ccc(Cl)o2)=O)CC2CCN(C(c3cc4ccccn4n3)=O)C2C1 N1(C(CCN(C(c2c[nH]c(=N)o2)=O)C2CC2)=O)CCC(O)CC1 N(C1CCCc2sc(Cl)cc21)c1ncnc(NCCCOC)c1C C1(NC(C(C)SCC)=O)CCCCN(C(c2nc(C)c(N)cc2C)=O)CC1 N1(C(CC2CCC(NC(C(C)(C)N3CCCC3)=O)C2)=O)CCC=C(F)C1 C12(C(=O)NCCCN(C(C3C(C)(C(=O)O)C3)=O)CCO)CC(C(F)(F)F)(C1)C2 C1(C(N2CC(CNC(c3cnn(C(C)C)c3N)=O)C2)=O)(OCC)CCCCCC1 C12(NC(C(C(C)C)F)=O)CC(CNC(c3cnn4c3CCCC4)=O)(C1)OC2(C)C C=CCC(C)(CC)C(=O)N1CCC(CCNC(=O)CCC2(C#N)CCC2)C1 C(=O)(CC(O)C(Cl)(Cl)Cl)N1CCC(NC(c2cc(C(C)C)c(N)cc2)=O)C1 CN1CCN(C(C2COCCO2)=O)C(CNC(c2cc3occc3[nH]2)=O)C1 O=C(N=c1[nH]oc2c1CCCC2)NCc1cc(Cl)c(F)cc1F N1(CC)CCN(C(c2ccc(OC(F)F)cc2C)C(=O)NC2CCOC2)CC1C C(c1cc(C)no1)=CC(=O)NCC1(CCNC(c2c(CCC)nco2)=O)CC1 CCC(CCC(=O)N1CC=CC1COC)NC(=O)CCCCCF C(=O)(C(CCc1ccsc1)NC(=O)OC(C)(C)C)N1CC(O)(CNC(=O)OC)C1 C1(C)(CC(=O)NCCOCCN(C)C(C2CCCCO2)=O)CC(F)(F)C1 CCC(O)(CC)c1cn(CCCC(=O)N(CC(=O)OC)CCN(C)C)nn1 c1(C(=O)NCCC2CCC(NC(C3(C=C)CCC3)=O)C2)coc2ccc(C)cc12 N1(C(COC2(C)CCC2)=O)CCC(C2CC2)C1C(=O)Nc1cnc(C2CC2)[nH]1 N1(C(c2c(SCC)cncc2)=O)CCC2(CCC2NC(C2CCCO2)=O)CC1 N#CC1(C(=O)NCC2(C(F)F)CCN(C(C3(n4cccn4)CC3)=O)C2)CC=CC1 N1(C(=O)OC)CCCC(N(C(CNC(=O)C=C2CCC2)=O)C)C1 C#Cc1ccc(Cl)c(C(=O)NC2(CNC(=O)C=Cc3sccc3C)CC2)c1 c1(C(=O)NC(C2CCN(C(=O)COCCCF)C2)C)cccc(-n2cncn2)n1 Cc1oc(C(=O)NC(C)CCNC(C2CCCCC2O)=O)cc1-c1ccccc1 Cc1cccc2c1OC(C(=O)NC1CC3(NC(=O)C4=CCCCO4)COC1C3)C2 S(=O)(=O)(c1nc(N2CCN3CCCC3C2)ccc1Br)NCCCC(C(C)C)O c1(C(=O)NC(CNC(c2c(OCC)oc(C)n2)=O)CO)cccc2c1COCC2 c1(CN=c2scc(CC(N3CCC(OCCF)C3)=O)[nH]2)cccc2c1OCCO2 c1(C(=O)NC(CN(C(=O)C(O)C(F)F)CC)C)cc(O)ccc1OC c1(C(C)NCc2ccc(OCC)cc2)ccccc1[N+](=O)[O-] N1(C(C2(Cl)C=CC(OC)=C2)=O)CCN(C(C2(OC)CCCOC2)=O)CC1C c1(C(=O)NC2CC(C)N(C(c3ccns3)=O)C2)c(F)cccc1Cl C1(NC(c2c(C)nsc2)=O)CCN(C(=O)C(C)NC(C2CCC2)=O)C1(C)C c1(C(=O)NCCOCCCNC(C(C)OCCCC)=O)cn2cc(C)nc2s1 C1(CC)C(NC(=O)C(F)CC2CCOC2)CCCN1C(C1CCOC1)=O N1(C(CCOCCN(C(C2(C(C)=O)CC2)=O)C)=O)CC2CCCN2CC1C NC1(NC(=O)NCc2ccnc(OCC(F)F)c2)CC(F)(F)C1 N1(C(c2cc(O)c(F)cc2N)=O)CCC(C=O)=C(F)C1.CO C(C)(N(C)N1CCC(C)C1)c1ccc(C)s1 CC1CCN(C(c2cc(F)cnc2O)=O)CCN1c1nc(C(C)(C)C)nc(=N)[nH]1 C(=O)(C(C)(C)C(=O)N1CCC(NC(c2cc(O)ncn2)=O)C1)OCC S(=O)(=O)(c1cccc(CN2C(=O)CCC2=O)c1)NC(C1C(C)CC(=O)N1)=O CN1CCn2ncc(COCc3nc(C4(F)CCOC4C)no3)c2C1=O c1(C(N2C3CN(C(c4cc(N)c(F)cn4)=O)C(C3)C2)=O)cnc2ccnn2c1 N1(C(C23N(C(C4=CCCC4C)=O)CCC2C3)=O)CC2(C1)CN(C)CCO2 Cc1c(C(=O)NC(C2CCCCN2C(=O)CCc2cn[nH]c2)C)nnn1C N1(C(COc2c(OC)cccc2)=O)CC(NC(c2cnnn2CC)=O)CC1(C)C CC(C)(CO)C(CNC(=O)NCCC(F)F)c1ccccc1 C1(C(N2CCC(CN(C(CCSC)=O)C)CC2)=O)Cc2ccccc2S1 C=CCCCCCCCC(=O)NC1CS(=O)(=O)CC1NC(C1CCCCC1)=O C(=O)(CC(C)(C)Cc1cn(-c2ccc(Br)c(C)c2)nn1)NCC(CC)C N1(C(c2cc(C)c(C)nn2)=O)CCC(NC(C2CN(C(C)C)C2)=O)CC(O)C1 Cc1ncc(CC(=O)NCCOC2CCN(C(=O)CC(C)N3CCCC3=O)C2)s1 Cc1cc(N)cnc1C(=O)N(CCCN(C)C)CCNC(=O)CC1CCCOC1 N1(C(C2CC(C)(CC)C2)=O)CCN(C(=O)C(C)SC(F)(F)F)CC12CC2 C1(C(C)=O)(Nc2ncnc(O)c2Br)CCN(C(c2cc(Cl)ccc2C)=O)CC1 C1(CNC(CC2CC(N(C)C)C2)=O)N(C(=O)Cc2ccccn2)CCCC1(C)C c1(C(N(C2CN(C(=O)C(C)(C)c3ncco3)CC2F)C)=O)cc(Cl)cnc1O C1(C(=O)NC2C(CC(=O)NCCC(C(C)C)C)C(O)C2)C2CCC(C2)C1C C1(CNC(CCC(=C)Br)=O)C(C2CC2)CCN1C(c1cnc(C)c(N)c1)=O c1(N2CCCC(OCC)C2)ccc(Br)c(S(=O)(=O)NC(c2cc(C)nn2C)C)n1 n1(CC(=O)NC2(COC)CCN(C(c3c[nH]cc3C)=O)C2)cc(P(C)(C)=O)cn1 C1(CCC)(NC(COCCC#C)=O)CCCN(C(=O)CC(C)C(=O)OC)C1 c1(OC)cc(C(=O)NC2CCN(C(c3cnco3)=O)C(C)C2)cc2cn(C)nc12 Nc1c(C(=O)NC(CNC(c2cc(F)ccc2F)=O)C2CC2)cc(Cl)cc1Cl C(=O)(CCCC(=O)NCCC1CCCN(C(=O)C=CBr)CC1)NCCC c1(C(=O)NCC2CC(NC(CC(CC)O)=O)C2(C)C)cnc2ncnn2c1C C1(NC(c2cnc(C)n2C)=O)CCN(C(C2(CN(C)C)CC2)=O)CC12CCC2 c1(N(C(CNC(C)C(c2ccccc2)O)=O)CCC#N)cnn(C)c1 c1(C(CO)NC(C(C)(C2CCOCC2)OC)=O)ccc(Cl)cc1 C(=O)(C1=NOCC1)N1C(C(=O)NCC2CCCCC2)CCC1 N1(C(C(c2ccc(C)cc2)C)=O)CC(NC(c2c[nH]nc2F)=O)C(N=[N+]=[N-])C1 c1(CC)cccc2[nH]c(C(N3CCC(CNC(C4CCO4)=O)C34CCC4)=O)cc12 C(N=c1[nH]c(-c2ccc(Br)nc2)cs1)c1cc(Cl)sc1 Cc1ccccc1C(C(=O)O)N(C)C(c1ccc(C2CCCOC2)cc1)=O C1(C(=O)CCC2(CNC(N)=O)CCCC2)CN(C(C23CCC(C2)C3)=O)CCO1 C12(CNC(c3n(CC)nnn3)(C)CCc3cccc4c3CC4)CC(C1)C(C)(C)O2 C1(C(=O)Nc2cccc(NC(C(c3n(C)cnc3)O)=O)c2)CCCC(C)(C)CC1 N1(C(CCN(CC(C(C)C)C)C)=O)CC2(C1)SCCC2NC(=O)CNC=O c1(OCC(=O)NC(C2CN(C(C3OCCO3)=O)CCO2)C)cc(Cl)cc(Cl)c1 c1(C(=O)NCC2(CNC(CC(=C=C)C)=O)CCOCC2)cc(C2CC2)nc(O)c1 C1(c2nnnn2CC2CCOCC2)(NCC2(C)COC2)CCN2CCCCC2C1 C(=O)(CC=C(Cl)Cl)NC(C(=O)NC(COCC)C)C1CCC1 C(C(F)(C(=O)NCCc1nncs1)C(C)C)NC(C(C)(C)NC(=O)OC)=O N1(C(C2CCOC2)=O)CCC2(CC1)CC2NC(C12COCC(C1)C2)=O CC(CC(F)(F)F)C(=O)NCC1CCN1C(C1CCC(C)(C)C1)=O N1(C(CC2C(=O)NC(=O)N2)=O)CC2(CC(NC(=O)C(F)(F)CO)C2)C1 C1(NC(c2cnc(C(F)F)[nH]2)=O)CN(C(C2CC2CF)=O)CC1C1CC1 N1(C(C=CC(C)=O)=O)CCC2(CCN(C(=O)C(C)(C)S(=O)(=O)C3CC3)C2)C1 N1(C(c2n(CC)ccn2)=O)CCN(C(C2(C(=O)N(C)C)CC2)=O)CC1C(C)(C)C N1(C(N2C(c3c(C(=O)O)c[nH]n3)CCCC2)=O)CC2(CC(O)C2)C1.c1ccns1 c1(C(N(CCCCCNC(C(C)N(C(C)=O)C)=O)C)=O)cc(Br)cnc1C c1(C(=O)NC2CC(NC(c3nn(C)c(O)c3)=O)CC2O)cc2cccnn2n1 C(=O)(CC(C)(C)C(F)F)N1CC(O)(C(C)NC(=O)C=Cc2ccc(Cl)s2)C1 c1(C(COC)NC(=O)Cc2cn(C3CCCNC3=O)nn2)cc2ccccc2s1 c1(OC)c(C)cc(-c2csc(NC(=O)C(C)(C)C(N)=O)c2)cc1C C1(NC(CCc2nnc(C)n2C)=O)CC12CCN(C(C1COC(=O)N1C)=O)CC2 CC1CCCc2c(C(N3CCCCC3CNC(C3(C(C)(F)F)CC3)=O)=O)cnn21 c1(C(C(=O)N2CC(Cn3cc(CCCCCO)nn3)C2)(F)F)ccc(F)cc1Cl c1(C(C)OC(NOCCCC(=O)OC(C)(C)C)=O)cc2c(s1)CCC(C(C)C)C2 C1(CNC(C(C2CCN(C(C3(F)CC=CCC3)=O)CC2)C)=O)CC2CCCC2C1 S(=O)(=O)(c1cc(C(F)(F)F)cc(Br)c1)NC(CCCC)(C)C(N)=O N1(C(CCC(N)=O)=O)CC2CCCC2(NC(c2cn(CC3(C)COC3)nn2)=O)C1 C1(CC)CN(C(=O)CCc2cc(C)no2)CCC1NC(=O)Cc1n[nH]c(=N)s1 c1(OC)cc(C(C)Nc2cc(C(=O)O)c(C)c(Br)c2)c(F)cc1F C1(NC(C=CC)=O)CCCCC1CNC(=O)CCCN1CCCC1 C(=O)(C1CCCn2cc(C)nc21)NCC1C(NC(Cc2cn(CC)nc2)=O)CC1 c1(C(=O)NC2CN(C(c3cnc(CCC)s3)=O)C(C)C2)cc(CC)ccc1N N1(CCC)CCCCC1C(N1CC(=O)CC1C(=O)NCCOCCOC)=O CC1(C)CC(C)(C(=O)NCCOC(C)(C)CNC(=O)CCC2CC2(Cl)Cl)C1 C(C)(CC(=O)NCC(C)(C)CNC(=O)C(F)(F)c1cnn(C)c1)OC Cn1[nH]c(C(=O)NCC(C(C)(C)C)NC(=O)CC2CNC(=O)C2)nc1=O c1(C(=O)NC2CCCN(C(c3c(C)noc3)=O)C2)n[nH]c2c1CCSC2 C#CC1CCCN(C(=O)C(F)CC2CN(C(C3C(=C)C3C(=O)OC)=O)C2)CC1 c1(NC(=O)NC2CN(C(C)=O)CC2N=[N+]=[N-])c(Cl)nc2ccccn12 N1(C(c2n(C)c(C3COCCN3C(=O)C(Cl)Cl)cc2)=O)CC(=O)N2CCCC2C1 N1(C(=O)NC(c2nnc3n2CCC3)C)CC2(CCCC2)c2c(F)cccc21 C1(C(=O)NC2CN(C(CCc3ccc(CC)cc3)=O)CC2C)CC(C)(C)CN1C c1(C(=O)NC(C(C)NC(C(CCCC)C)=O)C)cc(C)c2ncccc2c1 Cc1cc(C)c(CC(=O)NCC2CCN(C(=O)CC34CCC(CC3)C4)C2)c(O)n1 c1(N(CC)CC2CCN(C(C3CC(O)C3)=O)CC2)cc(C(C)C)nc(Cl)n1 CC1(C(N2CCC(O)C(NC(=O)C=CCF)C2)=O)CCCCCC1 CC1CCCN(C(c2n[nH]cc2CNC(C2CCNC(=O)C2)=O)=O)C1CO C(C)(C(CO)NC(C1CCS1(=O)=O)=O)NC(C(C)NC(C)=O)=O c1(CC)cncc(C(N2CCC(COC)C2)C(=O)NCCOCCC2CC2)c1 c12nc(=N)[nH]cc1C(=O)N1CCCC1C1CC1NC2.C(=O)(CCOC1CC1)OC C(=O)(C(C)(CO)NC(=O)CSC(C)C)N(CC(CCC)O)C Cc1ccc(O)cc1CNC(=O)CC(O)CNC(=O)C(C)C(C)(C)C CCC(CNC(C1(N(C)C)CCCC1)=O)(CC)C(=O)NC1CC(C)OC1=O N1(C(C2(CC)CCOC2)=O)C(CO)CSCC1c1ccccc1 c1(C(=O)NCC(CNC(C(CC=C)OC)=O)(C)F)cccc(O)c1F C1(C(N2C(CN(C(c3nc(CC)sc3N)=O)C)CCC2)=O)CCCCC12CCC2 c1(CC(=O)NC(c2scc(C)n2)C2CC2)ccc(Cl)cc1Br c1(NC)cccc(C(=O)N(C)CC2CCCN2C(c2csnc2Cl)=O)n1 C12(C(N(C(CC)CNC(c3ccc(C)c(C)n3)=O)C)=O)CCCCC1C2(F)F c1(C(=O)NCC2OCCN(C(c3cc(CC)sc3)=O)C2)ccc(F)c2[nH]ccc12 n1(CC2(CCNC(C3CC34CC4)=O)CCC2)cc(-c2c[nH]nc2C(F)F)nn1 C1(CNC(C(C)n2ccnc2)=O)CCC12CN(C(=O)Cc1nc([N+](=O)[O-])n[nH]1)C2 c1(C(=O)NC2C(C(N(CCC)CCC)=O)CCC2)cc(Cl)cnc1OC Cc1ncncc1C(N1CC=CC1C(=O)NCC(C)O)=O C12(C(=O)NCC(C)N(C)C(c3cnccn3)=O)CC(C(F)F)(C1)C2 C1(C(=O)NC(C)(C)C=CC(=O)NCC=C2CCSCC2)CCCCC1 C(CN=c1nc2sccc2c(NCC2CCC(O)CC2)[nH]1)(C1CCCC1)OCC c1(C(C)(C)O)ccccc1OCc1cc(C(C)(F)F)ccn1 CCCC(CC)C(=O)N1CCN(C(C2(C)CCN(C(C)=O)CC2)=O)CC1CCO C1(NC(CC(=C)C)=O)CC(C2CCN(C(c3cc(O)ccc3F)=O)C2)C1 C1(C(N(C(C)CCO)C)=O)CC2(CC(NC(c3ccno3)=O)C2)C1 C(=O)(CS(=O)(=O)CCO)NC1CCN(C(c2[nH]c(=N)sc2)=O)CC1F CC(C)C(O)C(F)(F)C(=O)NCC(C1CC1)N(C)C(C1(CCF)CCC1)=O C1(NC(C(CC#C)(C)C)=O)CN(C(=O)CC(C)CN(C)C)CC1N=[N+]=[N-] CN1CCN(CC(=O)NCC2(CO)CCN(C(c3cnc(Cl)s3)=O)C2)CC1 N1(CCNC(=O)CCc2cccnc2)CCN(C(=O)CNC2CCCC2O)CC1 N1(C(C2CC(=C)C2)=O)CCCC(CC)(NC(c2cc(C#N)oc2C)=O)C1 C1(N(C(c2c(C)cc(C)nc2)=O)C)CCN(C(C2C3CCCC23)=O)CC12CC2 C1(C(=O)NCc2c(OC)cccc2)CN(C(=O)CCC2CC2(F)F)C(C)(C)C1 C1(NC(C2CCC(C)C2)=O)CC1C1CCCN(C(c2cc3sccc3s2)=O)C1 C1(CNC(C2C(C)(C)C2(C)C)=O)CCCCN(C(=O)CCn2cnnn2)C1 Cc1nc(NCC(O)CNC(=O)Cc2ccc(O)nc2)c2c(C)csc2n1 C1(CC(=O)N(CCNC(c2csc(COC)n2)=O)CC)CCC(=O)N1C C1(CNC(CCCCC)=O)CCC(C)N(C(c2cn(CCO)nn2)=O)C1 C12(COC)CC(CNC(c3cccc(O)n3)=O)(CN1C(C1CC1CF)=O)C2 c1(C(N2CC=CC(NC(C3(CC#C)CCCO3)=O)C2)=O)cncc2sccc12 C1(C#N)(C(N(CC(C)(C)NC(C(CC)NC(C)=O)=O)CC)=O)CC2CC2C1 c12ccc(cc1)CC2=O.n1(CCOCC(=C)C)cc(C(C)(C)O)nn1.OC C(=O)(C1=CS(=O)CCC1)N(C1CCCN(C(=O)CCC2CCC2)C1)CC C1(CNC(c2cc(OC)n[nH]2)=O)CC2CCC1N2C(=O)CCc1ccsc1 Cc1nc2ncc(C(=O)NC3CCN(C(c4cc(F)c(N)c(F)c4)=O)C3)cc2o1 C1(NC(C(C)NC=O)=O)CN(C(=O)Cn2cccnc2=O)CC12CCCC2 C1(O)(CC)CCC(NC(C2(C)C=CCN2C(C2CC(C(=O)OC)C2)=O)=O)CC1 CC1CNCC(CN2CCC(F)(C(=O)N(C)C)C2)C1 c1(OCCC(=O)NCCC2CN(C(C(CC#C)C)=O)CC2C)ccc(F)cc1F N1(C(c2c(C)onc2C2CC2)=O)CC(NC(c2ccncc2O)=O)C2(CCC2)C1 Nc1ccc([N+](=O)[O-])c(C(N2CC(OCCNC(=O)CCC3CC3(F)F)C2)=O)c1 C1(NC(C2(C)CCCOC2)c2nnnn2CCOCC2CC2)CC1C1CCOCC1 N1(C(C(C)=CC2CC2)=O)CCCC(C)(C)C1CNC(C1CC12CCCCC2)=O CCCC(C(=O)N(CC(C)C(C)C)C)NC(C1(O)CCOC1)=O CC(C)C(C)(O)CNC(C1(C(C)NC(C2COC(=O)N2)=O)CC1)=O C(=O)(CC(F)(F)C(F)(F)F)NC1CCN(C(C(COC)COC)=O)CC1(C)C Cc1ncc([N+](=O)[O-])n1CC(N1CCC2(NC(=O)Cn3cnnn3)CC2C1)=O C(=O)(C1=CCOCC1)N(CC)CC1CCCCN1C(=O)CCCN(C)C n1(-c2ccoc2)nc(Cn2cncn2)nc1C1COCC1C1CC1 c1(C(=O)NC2CCN(Cc3ccc(COC)o3)C2)nc(OC)cc(OC)n1 C1(C(CC)NC(c2cnc(C3CCCC3)nc2)c2nnnn2C)CCCCCC1 c1(OCC)ccc(C(=O)O)cc1NC(C1(C)N(CC(=O)NC(N)=O)CC1)=O Cc1nn(C)c(-n2cncn2)c1CN(C)Cc1n[nH]c(-c2ccccc2)c1C N1(C(C2N(C(C)C)CCC2)=O)CCN(C(c2c[nH]cc(Cl)c2=O)=O)C(CF)C1 C(=O)(C(C)S(N)(=O)=O)N1CC(CCC)C(NC(c2ccc(OCCF)cn2)=O)C1 C(=O)(C(F)C(F)(F)F)NC(C(=O)NC1(C2CC2)CC1)Cc1ccco1 c1(OCC)ncnc(OCC)c1C(N1CCC(NC(C2(F)CCCOC2)=O)C1)=O N1(C(c2[nH]c(=NCc3c(C)cc(Br)cc3)sc2)=O)CCC2(CC1)CN(C)CCO2 N1(C(=O)COC2CCS(=O)(=O)C2)CCN(C(C2C3CCC2CC3)=O)C2CCC12 C1(C)(OC)CC(NC(C23CC2CCN3C(c2ccc(N(C)C)nn2)=O)=O)C1(C)C c1(C(=O)NC(C2CCN(C(c3c(C)cc(CC)o3)=O)C2)C)ccnc2[nH]cnc12 Cn1nc(C(=O)NCCC2(NC(C3CC4C=CC3O4)=O)CC2)c(Br)c1Cl c1(OC)cnc(C)cc1-c1cnc(C2CCCN2C(C2CC2C2CC2)=O)[nH]1 CN1CCCC(C)(C(N2CCC(CN(C)C(C3CC4(CC4)CO3)=O)C2)=O)C1 N1(C(C=COCC)=O)CCOCC1CN(C(=O)C(n1nc(C)cc1C)C)C C(=O)(C1=CS(=O)(=O)c2ccccc21)NCC1N(C(C2N(C=O)CCC2)=O)CC=C1 Cc1ccc(C(=O)NCC2CCCN(C(C3CCC(F)(F)C3)=O)C2)cc1 c1(C(N2C(c3nc(CC)sc3)CCC2)=O)cc([N+](=O)[O-])oc1C S(=O)(=O)(c1cccc(N(C)CC2CC2c2ccnn2C)n1)N(CC(CCC)C)C Cc1nc(=N)[nH]c(=NCC(C)N(C)C(C2CC(C)(C)CC(C)(C)C2)=O)[nH]1 c1(C(=O)NCC(C)(C2CC2)NC(C(=Cc2cccs2)C)=O)cncc(O)c1Cl CC(=O)CCCC(C)C(=O)NC(C(=O)NC(C)C(C)(C)C)C1(O)CCC1 C(=O)(C(C)(C)C(=O)NCC(CO)NC(c1sc(C)c(Br)c1C)=O)OCC Cn1cnn(CC(=O)N(CCC(=O)NCc2ccccc2)C2CCC2)c1=O Cc1ccnc(N2CC(=C(F)CNC(=O)C(C)(O)C3CCC3)C2)c1[N+](=O)[O-] C1(C(=O)NC(CC)CNC(=O)CC2CC2(Cl)Cl)CC12CCOC2 c1(C(N(C2CN(C(=O)CNC(=O)NC3CC3)C2)C)=O)ccc(-c2ccncc2)s1 C1(C2CCCOC2)(NC(C2C(CNC(C3(C)CC(=C)C3)=O)CCCC2)=O)CC1 N1(C(C2OCCN(CC)C2)=O)CC2(CCN(C(=O)CCc3ccncn3)C2)C1 C(CC(=O)NN1CCCC1C(=O)NCC1(C(N)=O)CCC1)=CC(C)(C)C c1(C(N2CCN(C(c3c(CC)ocn3)=O)C3C2C3)=O)cc(C)cc(F)c1N C1(CN(c2n(CCCOC)c(-c3ccc(C#N)[nH]3)nn2)C)C(F)(F)C12CCCC2 CCC(CC(=O)NC(CNC(C1CCC(F)(F)C1)=O)C1CCC1)OC c1(CCC(N2CCC(O)(CNC(CCC(C)O)=O)C2)=O)ccnc2ccccc12 C1(NC(c2c(C)[nH]nc2Cl)=O)CS(=O)(=O)CC1NC(C1(n2nccn2)CC1)=O N1(C(C2C(NC(=O)C=Cc3cccnc3)COC2)=O)CCC(C2CCC2)C1 c1(CC)cnccc1OC.c12cnn(c1)CC(=O)NCC(C)(C)CN(C)C(=O)C2 N1(c2ncc(C)cn2)CCCC1C1CCCCN1C(c1cccn2nccc12)=O c1(NC(C2C(NCc3c(OC)cncc3)CCCC2)=O)cccc2c1OCCO2 C=CC(CCC)CC(=O)NC1CCC(N(C(=O)C(COC)N(C)C)C)CC1 N1(C(Cc2cn(C3C(OC)COC3)nn2)=O)CC(C(=O)OC(C)(C)C)C2(CC2)C1 c1(C(N2CCC(CC3CCCCC3)CC2)C)ccc(C(N2CCOCC2)C)cc1 C1(NC(C(=O)NC2CC2)=O)CCN(C(c2cnc3[nH]cncc2-3)=O)C12CCCC2 C(c1ccc(Cl)cc1)=C(C(N1CCC(CN(C)C(c2cnco2)=O)CC1)=O)C#N C1(NC(C2C(C)(C)C2)=O)CCSC12CN(C(c1cc(O)cc(Cl)c1)=O)C2 c1(C(=O)NC(C2CCCN2C(=O)CS(=O)(=O)CCO)C)cc2c(=O)[nH]ccn2n1 C(N=c1[nH]c(=NCc2cc(C)ns2)[nH]c2cc(C)ccc12)C1C(C(=C)C)OCC1 N1(C(c2n(C(C)C)ccc2)=O)CC2CC1CC2NC(c1cccc(CO)n1)=O N1(C(c2c(CNC(C3C4CCC(=O)C43)=O)cco2)=O)CCC(F)(CF)CC1 c1(C(=O)OC)cc2cc(N(C)C(c3c(N)cccc3Br)=O)ccc2o1 C1(C(N)=O)(CNC(c2ccn(CCC)n2)=O)CC(F)(F)C1 C(=O)(CCC(C)(F)F)C(=O)CC1(NC)CC1.CC(CS(C)=O)NC c1(OC)cc(C(=O)NC2CC(CCNC(C3(C)CCC3)=O)C2)ccc1O c1(C(N2CC(CNC(C=Cc3nnc(C)o3)=O)N(C)CC2)=O)ccc(S(N)(=O)=O)s1 N1(C(CCCNC(=O)OCC)=O)CCC(NC(=O)CN(C)C(=O)OC)C(C)(C)C1 c1(C(N2C(C(C)NC(Cn3c(C)nc(C)n3)=O)CCC2)=O)cc2sc(C)cc2s1 c1(OC)cccc(C(=O)NC2CN(C(=O)CNC(c3cccs3)=O)C2)c1[N+](=O)[O-] Cc1cccc(C(C(C)C)N(C=O)Cc2cn(C)c(C)n2)c1 N12CCC3(CC1)CC3C2=O.Cc1cc(Cl)cnc1C(=O)Nc1ccc(N(C)C)nc1 N1(C(C(N2CCC3CC23)=O)=O)CCC(COC2CCCCC2)CC1 Cc1ccc(C(N2CC3(C)CC2(C(N2CCC(O)(C(C)C)C2)=O)C3)=O)cc1F C1(O)(C(C)NC(c2ccn(CCF)n2)=O)CCN(C(=O)CCOCC(F)F)C1 O=C1CN(C(c2coc(CNC(=O)CC=C(Cl)Cl)n2)=O)CC2(CC2)N1 c1(NC(c2cc(-c3ccc(C)nc3C)[nH]n2)=O)c(Cl)cccc1C#N c1(CC(N2CC(O)(C(C)NC(c3ccnnc3)=O)C2)=O)cnc2ccccc2c1 C=CCCC(F)(F)C(=O)NCc1ncoc1CCNC(C1CCCS1)=O CC(O)CCCCCC(=O)N1CCC2(CCCN2C(c2ccc(N)c(O)c2)=O)C1 C(C(=O)N=c1ccn(CCO)[nH]1)C1(C)N(C(COC2(C)CCCC2)=O)CC1 c1(CC)ccc(C(=O)NC2CC(CCNC(C3CCS(=O)CC3)=O)C2)c(F)c1 C(C(F)F)(C(C)(C)C)NC(CC(C)(C)N(C(c1cncc(OC)c1)=O)C)=O c1(C(N2CCC3(NC(Cc4c(C)occ4)=O)C(C2)C3)=O)cnc2ccnn2c1C c1(-c2c(C(N(C)Cc3nc(C)on3)=O)csc2)cnccc1C#N C(CC(C)C)(C(=O)N1CCCCC1)NC(c1scc(-c2cn(CC)nc2)c1)=O Cc1ccc(-c2cc(C(=O)NC3(C)CCN(C(c4cc[nH]c4)=O)C3)n[nH]2)cc1C Cc1cccc(C)c1C(O)C(N1CC2CC(NC(=O)Cc3nonc3C)C1C2)=O C1(NC(NCc2n(C(C)C)ncn2)=NCc2cnsc2)CCc2ccccc2C1 C(N=c1[nH]c(=NCC(C)(C)N(C)C)c2c(F)cccc2[nH]1)c1c(C)cc(Cl)cc1 C1(C(N2CC(C=C)(CC(=O)NCCC3(CO)CC3)C2)=O)CC(=O)C12CCC2 N1(C(C2C(=C)C2)=O)CCS(=O)(=O)C(CCNC(c2c[nH]c(C(N)=O)c2)=O)C1 C=CC1CN(C(c2cc(OC)ns2)=O)CC1NC(=O)C1=COCCO1 C1(CNC(C(=O)NCC)=O)CN(C(c2ccc(C(F)F)o2)=O)CC1O c1(C(N(C(C)C(N2CCC(CC)CC2)=O)CCC)=O)ccc2cncn2c1 C1(NC(C(C)NS(C)(=O)=O)=O)CCN(C(=O)C(c2ccccc2)C)CC1 S(=O)(=O)(c1ccc(C(=O)NC)cc1Br)N(CCC)CCNC1CC1C1CC1C C=C(F)C1(CC(=O)NCC(C2CC2)NC(C2(COC)CC2)=O)CCC1 N1(C(C2CC(OC)C2)=O)CC(C(=O)NCc2conc2C)C(C)(C)C1 C(=O)(C#CC1CCOCC1)NCC(C(C)C)(C)NC(c1ccc(Cl)[nH]1)=O CCCCC(C(=O)NCC(C)CNC(=O)CCc1ccncn1)C(C)C C(C)(C)(C(=O)NCC1CCCN1C(=O)C(C)c1ccsn1)SC c1(OCC(=O)NC2(C3N(C(COC)=O)CCC3)CC2)ccccc1CC(F)(F)F C12(NC(CCSC)=O)CCCC(CN(C(C3CCC(=O)N(C(C)C)C3)=O)C1)C2 N1(C(c2c(CC)ocn2)=O)CCN(C(C2CC=CC2)=O)CC1C(F)F Cc1nc(CC(=O)NCCOC2CCN(C(c3scnc3Cl)=O)C2)n[nH]1 C1(Cc2cn(C)nc2)CCN(c2ncc(I)cn2)CC1O c1(C(=O)NCC2C(CNC(c3cc(OC)nn3C)=O)C2)nccn2ccnc12 C1(CNC(c2cc(OCC)n[nH]2)=O)C(C)CCCN1C(c1coc(Br)c1)=O C=CCC(Cc1ccccc1)C(=O)NC(C)C(CO)NC(=O)Cc1sccc1C N1(c2n(CCC#C)c(-c3ccc(OC)o3)nn2)CCN(C)C(C)C1C N1(CCNC(C2C3CCC2(c2cscn2)C3)=O)CCN(C(c2ccsc2)=O)CC1 Cc1cc(C)c(C(=O)NC2CN(C(=O)Cc3cnn(C)c3)CC3(CC3)C2)c(O)n1 C1(CC)CCCC1C(=O)NCCN(C(c1ccc(C(=O)OC)o1)=O)C1CC1 C12(NC(c3ccc(C)n3C)=O)CCN(C(c3ccc(C(N)=O)cc3)=O)CCC1C2 C(=O)(CCC1=CCc2ccccc21)NCC(CCNC(C=CS(C)=O)=O)O N1(C(c2c(COC)cccn2)=O)CC2CCC(C1)C(NC(=O)C(C)CC1CC1)C2 c1(C(=O)NC2(CNC(C(CCC#C)O)=O)CCCC2)ccc2c(c1)COC2=O C(C(C(C)C(C)C)NC(c1cc(O)ncn1)=O)NC(c1c(C(C)C)ncnc1)=O c1(C(=O)Nc2ccc(C)c(NC(N)=O)c2)cc2c(Br)cc(F)cc2[nH]1 c1(C(C)C)ccc(C(=O)NC2CCN(C(=O)C(F)(F)C(F)F)CC2C)c(O)n1 c1(C(=O)NC2(C)CN(C(=O)CC3CCC(=O)O3)C2)cnn2c(=O)cc[nH]c12 CC(CNC(=O)C=C1CCCCC1)CC(=O)NOCc1ccccc1F CC(C)(CC(=O)N1CCC(C)(CCNC(c2coc(C(F)F)n2)=O)C1)C(F)F N1(C(CCN(C(c2c(Cl)cccc2Cl)C)C)=O)CCCC2(CCOC2)C1 C(=O)(C#CC1CC(F)(F)C1)NC(C)CNC(=O)CSc1cccc(F)c1 c1(C(=O)NC23CC(CNC(=O)CN4CCCOC4=O)(C2)C3)cccc2sccc12 C(=O)(C(C#N)C(C)(C)C)NC1COCC1N(C)C.c12cc[nH]c1C(=O)N(C)C2 c1(C(=O)NCC2OCC(CNC(COC(C)C)=O)C2)c(Cl)ccc2c[nH]nc12 c1(CC)nc(C(=O)NC2CCCC(CNC(=O)CC3CC=CC3)C2)c(N)s1 C1(C(=O)NCC(CNCc2ccnc(C)n2)O)COCCN(CC(F)(F)F)C1 c1(OC)ccccc1S(=O)(=O)N1CC2(CCN2C(=O)CN(C)C(C)C)C1 C(=O)(CC(CC)CCC)NCC(CCCC)NC(=O)Cc1ccc2c(c1)CCC2 C12(C(=O)Nc3c(C)noc3)CC(CO)(CN1C(C1CC(=O)C1)=O)C2 CCCCCC(=O)NCC(CC(C)C)NC(C1(C(N)=O)CCC1)=O C(CC(C)C)(C(=O)NC1CN(C(=O)CCC2CCCCC2)CC12CC2)OC c1(C(N2CCC(NC(c3ccco3)=O)CC2)C)ccc(F)cc1F n1(CC(=O)NCC2(C(N)=O)CN(c3nccc(CO)n3)C2)ccccc1=O C(=O)(CCCC(=O)N1CCC(O)(CN(C)C(c2c(Cl)csc2Cl)=O)C1)N(C)C CC1(C)C(CNC(=O)C=Cc2cccc(Cl)c2)CCN1C(C1CC2C=CC1C2)=O c1(OC)cc(Cl)ccc1-c1cc(CNc2cccc(OC(F)F)n2)[nH]n1 c1(C(=O)NCCCOCCNC(C2(C)CCOC2)=O)cc(Cl)c2c(c1)OCCO2 c1(SCC)ccccc1CC(=O)NC1CC(C)(NC(=O)C=CC(C)C)C1 C1(C(=O)O)CC2CN(C(=O)CC(C(F)(F)F)c3ccon3)CC2C1 CC1=C(C(=O)NCC2(NC(C3CC3C)=O)CCCCC2C)CCS1(=O)=O N1(C(COCc2cc(C)on2)=O)CCCN(C(=O)CC2CCN(C)C2)C(CO)C1 C1(C(=O)Nc2cccc(OCC)c2)CC(O)C(O)CN1 C(=O)(C(F)CC(C)(C)NC(c1cn(C)cn1)=O)NCC(C(=O)OC)(F)F c1(OCC)cnc(C(=O)NCC2CCC(NC(=O)C(C)(Cl)Cl)C2)cn1 N1(Cc2ccc(C3(C)NC(=O)NC3=O)cc2)CCC2(C1)OCC1CC21 CC(C)(O)C(F)(F)C(=O)NCC1(O)CN(C(=O)CCC2CCCOC2)C1 N1(C(C2(OCC)CCC2)=O)CC2CC(C1)N(C(=O)Cc1c[nH]nc1C)C2 c1(C(=O)OC)ccc(C2CCCN2C(=O)NCCn2nccn2)cc1 N1(CCCC(=O)NCCN(C(c2c[nH]cc2C2CC2)=O)CC)C(=O)CCC1=O C1(COC)CCN(S(=O)(=O)N2CCC(C)(OCc3ccc(OC)cc3)CC2)CC1 CC(C)(C#N)CC(=O)NCC(F)CNC(=O)C=CCCCCCCCO C(CCC(=O)NCCC(O)CNC(c1cnn(C)c1)=O)N(CCC)CCC CC#CCCCCN=c1[nH]c(=NC2CCN(C(C)=O)C2)[nH]c2c(F)cccc12 c1(OC)ccccc1C(C)C(=O)N(C)CCNC(C1(N2CCCC2)CCCC1)=O C1(CC(=O)NCCCc2ccccc2)CCN(C(=O)NC2CCSC2)C1 Cc1cc(CC(N2CC(C(N)=O)(CNC(=O)CN3CCCC(O)C3)C2)=O)n(C)n1 c1(CC)cnccc1C(=O)NCC1(C)CCCN1C(=O)CC1(c2ccon2)CC1 c1(C(N2CCC(NC(C(CC=C)C)=O)(CO)C2)=O)cc(Cl)cc(Cl)c1Cl CC1C(C)N(C(=O)CCF)CCN1C(=O)COC1(C)CCOCC1 Cc1nc2cncc(C(=O)NCC3CC3CC(C)(C)C)c2[nH]1 c1(CC(=O)NC2CCC2NC(c2cc(C3CC3)on2)=O)c(O)ncnc1O C1(CNC(C2(C#C)CC2)=O)(NC(=O)COc2c(C)nn(C)c2C)CCCCC1C C#CC1(CN(C)C)CN(CC(C2CC=CCC2CO)=O)C1 C(C)(CNC(c1cnc(OCC(F)F)cn1)=O)(CC(C)C)NC(C(COC)C)=O c1(CC)nc(=NCC2CNC(=O)c3ccccc32)c2ccccc2[nH]1 N1(C(C2(NC(c3ncccc3F)=O)CCCC2)=O)CCC2=C(CCCC2)C1 C1(C(N(CCC2N(C(c3nc(C)nn3C)=O)CCCC2)C)=O)C(C)(C)OC1(C)C C1(NC(C(C=C)CC)=O)CCN(C(c2cc(C)n(C)c2)=O)C(C)C1 CC1(C)COC(CCC(=O)NC2CCCCC2n2cc(-c3nccs3)nn2)C1 c1(OC)cc(N2CC3(CCC(C(=O)NC(C)(C)C)O3)C2)nc(S(C)(=O)=O)n1 C(CCCCCCC)NCC(N1CCC(O)(CC(=O)NC(C(C)=CCC)=O)C1)=O C(CC(C(=O)N(C)CC1CCC(=O)O1)NC(C)=O)SC C1(C2(O)CCOCC2)(C(=O)NCC2(CO)CCN(C(C(=O)NCC)=O)CC2)CC1 C(=O)(CC(O)CCSC)N1CC(NC(COC)=O)C(O)C1 N1(C(CC(=C)C)=O)CC2(CCC(NC(C3(C)CC3C(F)(F)F)=O)CC2)C1 C1(F)(C(=O)NC(CSCC)CO)CCN(C(=O)CC2CCCC3CC23)C1 Cc1c(C(=O)NC2CCN(C(=O)CC3C=CCC3)C2C)c(O)nc2ccccc12 N1(C(Cc2nnc(C)o2)=O)CCC(C)C1CNC(C1(F)CC1)=O c1(NCCN(CC(C)(C)C)CC)c(C)cccc1C N1(C(C2CC(F)(CF)C2)=O)CCCOC(CNC(C2(O)CC2)=O)C1 N1(C(C(=O)NCC)=O)CCCC(C2CCN(C(C3C4CC5C(C4)C35)=O)CC2)C1 c1(NCC(c2ncc(C)s2)C)cnc(Cl)nc1Br C(=O)(C(F)(CC)C(=O)OC)N(CC(CNC(C(CC=CCC)C)=O)(C)C)C CC1CCc2[nH]nc(C(=O)N(C3CCNCC3C)CC3CC3)c2C1 N1(C(c2c(CCC)nco2)=O)CCC2(CC1)CCN(C(=O)Cn1ncnn1)C2 Nc1cc(C(N2CCC(NC(C3CC3(F)F)=O)C23CC3)=O)cc(O)c1 N1(C(c2c(CC)cncc2)=O)CCC(C(=O)N(CC(N2CCCC2)C)C)C12CC2 C1(NC(c2c(C)c(O)ccc2)=O)CCCC12CN(C(=O)CCCN(C)C)C2 C1(CC)C(NC(c2cc(C(N)=O)c[nH]2)=O)CCN1C(=O)C(Cc1ccsc1)OC c1(NC(Cc2cc3cnn(C)c3cc2)=O)nc2n(c1C#N)CCOC2 CC1CC(C(=O)NCC2CCCN(C(C3CC34CCOC4)=O)C2)=NO1 N1(C(c2cccc(C)n2)=O)CCC(NC(=O)C(C)NC(C2CCC2)=O)CC1C C1(OC)CC(C)CN(C(c2c(C)noc2C)C(=O)NCCC2(C)CC2)C1 CCCCCCC(C)NC(=O)CCn1cc(-c2c(C)nn(C)c2Cl)nn1 C(C(C)(C)C(C)(C)C)NC(C(CC=CC)NC(c1cccc(F)c1F)=O)=O c1(NC(CSCCNC(Cc2ccc(C)o2)=O)=O)cccc(Cl)c1C Cc1cccc(N)c1C(=O)NC1CCC(N(C(=O)C2=CC(C)(C)C2)C)C1 c1(C(N2CC(C)(NC(CN3CCC(C)CC3)=O)C2)=O)c[nH]c2ccncc12 C1(NC(C2(C=C)CC2)=O)CCCN(C(c2cccc(C)c2OCC)=O)CCC1 N1(C(c2cc(C3CCOC3)[nH]n2)=O)CCC2(CCCN2C(=O)Cc2nc[nH]n2)C1 c1(C(N2CCC(N(C(c3cc(C)on3)=O)C)C2)=O)ccc(C2CCCO2)nn1 CC(CCC(=O)NC1CN(C(c2ccc(C(F)(F)F)cn2)=O)CC1C)N(C)C c1(C(=O)NCCC(C)NC(C2CC2C(F)(F)F)=O)csc(-c2ncc[nH]2)n1 N1(C(CCCCCC)=O)CCC2CCCN(C(c3cccn4nnnc34)=O)C2C1 CS(=O)(=O)c1ccc(F)c(COC(=O)CCCC2CCCCC2)c1 C(=O)(N1CC2COCC2O1)C1C2N(C(c3nccc(CC)c3)=O)C(CC2)C1 CCCCCCC(CC)(CC)C(=O)NC1CCC(CNC(=O)C2=CCSC2)C1 C1(C(=O)NCC(CCOC)O)CCN(C(=O)c2csnn2)O1 CC(C)C1=NOC(C)(C(=O)NNC(c2ccc(C(F)(F)F)cc2)=O)C1 C12(C(N(CC(F)F)CC)=O)CCC(CC1)N(C(c1c[nH]nc1Cl)=O)C2 C1(NC(c2c(C)con2)=O)CCCC(N(C(=O)CCCCN(C)C(C)C)C)C1 N1(C(c2c(C)occ2)=O)CC2(CC(CNC(C3CC3c3cnnn3C)=O)C2)C1 C(=O)(C(C)S(N)(=O)=O)N1CCC(C(=O)NC(CC)C(C)(F)F)C1 C1(C(C)NC(=O)CC2CC(NC(=O)CN3CCN(C)CC3)C2)CC2(CCC2)C1 Cn1c([N+](=O)[O-])cnc1C(=O)NCC(C)(O)CNC(c1cccc(N)c1F)=O c1(C(=O)NC2CC(CNC(C3(O)CCC(CC)C3)=O)C2)cc2c(=O)[nH]ccn2n1 C(C(C)(C)CNC(C1CC1C#N)=O)N(C(=O)C(=O)NCC(F)F)CC c1(OC)ccc(C(=O)NC2C=CC(CC(=O)N(CCCN(C)C)C)C2)nn1 C1(O)(CN(C(CN(CCC)C)=O)C)CCN(C(=O)Cc2cnc(C)[nH]2)C1 C1(NC(c2csc(C(F)(F)F)n2)=O)CC(F)(CNC(C2CCS2(=O)=O)=O)C1 CN1CCCC(Cc2nc(-c3cccc(F)c3)nn2CCS(C)(=O)=O)C1=O C1(CC)(NC(=O)Cc2cnn(CC)c2)CCCN(C(=O)CSc2ccncc2)C1 N1(C(C(C)N2CCC2)=O)CCC2(CC1)CN(C(c1c(C3CC3)cnn1C)=O)C2 c1(C(=O)NCC(CCNC(C2=CC(C)(C)C2)=O)O)cnc2[nH]ncc2c1 c1(CNC(=O)CNC(C2CCCC2NC(C=C(COC)C)=O)=O)cccc(C)c1 C1(C2CCCN(C(c3cccc(F)c3SC)=O)C2)(NC(CC(C=C)C)=O)CC1 n1(CC)nccc1C=CC(=O)NC1CC(F)(CNC(=O)C(C)OCCN(C)C)C1 c1(OCC)cncc(C(=O)NCCCN(C(=O)C(F)CC)C(C)C)c1 C1(N(C)C(c2cc[nH]c2)=O)CN(C(c2ccn(CC(F)F)c(=O)c2)=O)CC12CC2 N1(C(c2ncn(CC)n2)=O)CCCC(C2CCN(C(c3ccco3)=O)CC2)CC1 c1(C(N(C2CN(C(=O)C(F)(F)CO)CC23CC3)C)=O)ccc(C(C)(F)F)nc1O C1(NC(C2(CC#C)CCC2)=O)CN(C(c2[nH]ccc2C)=O)C(C)(C)C1 C1(NC(CN(C(=O)CN2CCNC2=O)CCOC)=O)CC12CC(O)C2 c1(C(N2CCC(N(C(c3cc(CC)ncc3)=O)C)C2)=O)cc(=O)cc(Cl)[nH]1 CC(C)C(C(C)NC(=O)CCC(=O)N(C)C)NC(=O)C(=O)NC1CC1 Cc1c(NC(=O)C(O)CCNC(C2CC(=O)NC(=O)N2)=O)cccc1Cl N1(C(C(CCC)CCC)=O)CC=C(C(C)(C)C(=O)NCC(=O)OCC)C1 CC1CCN(C(C2CCCC(O)C2)=O)CCN1C(c1ccc(CN=[N+]=[N-])o1)=O N1(C(=O)CC2CCCOC2)CC(O)(C(F)F)C1.N12CC(C1)CN(C)CC2=O C#Cc1c[nH]nc1C(N1CCC(F)(C(=O)NCCc2nnc(C)n2C)C1)=O N1(C(C2CCOCC2)=O)CCC2(CC1)CC2(CO)CNC(C1(C(F)F)CC1)=O c1(C(N2CCN(C(c3ccn(C(F)(F)F)n3)=O)CC2)=O)ccc(O)c(F)c1F N1(C(C(CC(C)C)C)=O)CC(NC(=O)CCCSC(C)(C)C)CC2(CC2)C1 C(=O)(C1CCCc2nc[nH]c21)N1CC(n2cc(-c3c(C)ccnc3)nn2)C(O)C1 N1(C(C(C2CC2)OCC)=O)CC(CC(N2CCC(C#N)C2)=O)C(C)C1 c1(C(N(C)CC2(NC(CC(CC)C(F)F)=O)CC2)=O)ccc2cccc(Cl)c2n1 N1(C(C(N2CCCC(O)(COC)C2)=O)=O)CCOC2(CCN(C)C2)C1 C(=O)(C(O)C(C)(C)C)NCC(CNC(c1ccc(C)nc1C1CC1)=O)OC N1(C(C2N(C(c3n(C=C)ncc3)=O)CCCC2)=O)CCOC(C)CC1 C(=O)(C1=C(C)CCOC1)NC(CCCNC(c1ccc(OCCC)c(N)c1)=O)C N1(C(C)CNC(c2cccnc2)=O)CCN(C(C2CCC(=O)N2)=O)CC1 N1(C(C2CN(CC)C(=O)C2)=O)CCOCC(NC(C2C=CCC2)=O)C1 Cc1ccc2c(=NCCOc3ccncc3)[nH]c(N3CCC(C#N)C3)nc2c1 N1(C(c2nc(CCCCC)oc2)=O)CC2CCN(C(=O)CC3CC(C)=NO3)C2C1 N1(C(c2cc(C)n(C)n2)=O)CC2(CCC2)CC1C(=O)N(C)OCc1ccccc1 C1(C(=O)NCC(c2ccc(C)cc2)NC(c2ccco2)=O)CCc2cncn2C1 c1(C(=O)NC2C(CC)CN(C(c3cn[nH]c3)=O)C2)ccc(-n2cccn2)c(C)c1 C1(CCNC(C(C)(C)Oc2ccccc2)=O)CCCCN1C(c1csnn1)=O C(=O)(CCCC(F)(F)CO)N1CCCC(CN(C(C2C(C(C)C)C2)=O)C)C1 Cn1nnc2cc(C(N3CCN(C(c4ccc(O)c(F)c4)=O)CC(O)C3)=O)sc12 Cc1cc(C(=O)NCC2(CCNC(=O)CC3(C(F)F)CC3)CC2)n(C)n1 c1(C(N2CCCC(C(C)(C)O)C2)C(=O)NC(CC)C)cccc(C)n1 C(=O)(CCC1=CCCCC1)NC1C(NC(c2cc(C)nc(N(C)C)n2)=O)COC1 C(=O)(CC(C)(C)C(C)(F)F)N(C1CCN(C(CS(CC)=O)=O)C1C1CC1)C1CC1 c1(C(C)C)cc(C(=O)NCC2CC(F)(CNC(=O)CC3CCC4CC34)C2)nn1C N1(C(c2scc(-c3c(OCCC)cccn3)c2)=O)CCCc2ccc(OC)cc21 c1(-c2cn(C)nn2)nnc(N2CCCC2)n1CCC1(O)CCCC1 N1(C(CC2CC(CC)C2)=O)CCCC1C(C)NC(=O)COc1cn[nH]c1 c1(C(c2nnnn2C)NCCCOC(C)=O)ccc(OCCO)cc1C C1(NC(C(CC#C)C2CC2)=O)CCCN(C(=O)Cn2nc(C)nc2C)C1C C(=O)(C(CC(F)F)NC(C1CCC(F)(F)C1)=O)NC(CCC=C)C1CC1 C1(C(C(=O)CCOC(=O)C(C)CC2CCCCC2)=O)CCC(=O)C(O)C1.CCO N1(C(C(CC)OC)=O)CCC(C)C(NC(=O)CCCCCNC(N)=O)C1C O=C1CS(=O)(=O)CC(C(=O)NCc2cn(C3CCN(C(=O)C=CCO)CC3)nn2)N1 C(CN(C)C(C1CCCN(C)C1)=O)(CO)(CO)NC(CSCC=C)=O C1(CCNC(=NC)NC2CCN(CCc3ccccc3)CC2)CC(=O)N(C)C1=O Cc1ccc(C(N2CCN(C(=O)C(c3ccc(Cl)cc3)C)CC2)=O)c(N)c1Cl N1(CC)CCCC1C(=O)NC1CC(CC(=O)NC(C)CCC=C(C)C)C1 c1(CC)cc(NCC2(O)CN(C(=O)COCC(N3CCCC3)C)C2)ncn1 C1(C(N(CC(CNC(C(C(C)C)OCC)=O)(C)C)CC)=O)CCCCC1(F)F N1(CC(N2CC(CC(=O)OC)C(C)C2)=O)CCC(c2ccccc2)NC1=O c1(SC)ccc(CN(C(=O)C(F)CC2CCCCC2)C)cc1 C(=O)(C(C)CC(C)(F)F)NCCC1CCCN(C(CCC(=O)N(C(C)C)C)=O)C1 C1(NC(CSc2c(OC)cccc2)=O)CCCCN(C(C23CCC2C3)=O)C1 c1(C(=O)NC23CC(NC(C(CSC)OC)=O)(C2)C3)nc(C)ncc1Br C(CCCCCCO)NC(C(CC1CCC1)NC(C(CC)C)=O)=O N1(C(C(CC)C)=O)CC2(CCN2C(=O)C(CC)C(=O)OC)C1 C#CC1(O)CCN(C(c2noc3nccnc23)=O)CC1.C1C(=O)N1 C1(NC(c2cncc(OC)c2)=O)CN(C(=O)C(C)C(F)(F)F)CCC1(C)C C1(N(C(C(CC)C2CCOCC2)=O)C)(C(=O)O)CCC(c2cn(CC)nn2)CC1 CC(C)C(C)C(CNC(=O)C=C1CCN(C)C1)NC(c1cc[nH]c1)=O C1(C(=O)NCCCOCCNC(=O)C(F)=C2CCC2)OCC2COCCC12 C1(CC=C)(NC(=O)Cc2cnnn2C)CCN(C(c2ccc(Br)o2)=O)C1 c1(N2CCC(=CC(=O)Nc3cncc(C)n3)CC2)ncnc2c(Br)cccc12 c1(OC)cc(C(=O)NCC#CCNC(=O)C(C)(C)F)ccc1O.C1(CC2CC2)CC1 C(=O)(CCC(C(=O)NCC1CCC1NC(=O)COCP(C)(C)=O)N(C)C)OC C#CCC(CC#C)C(=O)N(CC(C)NC(=O)CC(C(N)=O)NC(C)=O)CC N1(C(C(C)Oc2ccccc2)=O)CCC(O)(CNC(C2(C)CCNC2=O)=O)CC1 C(=O)(C(C)(C)CNC(C)=O)NCCCCCNC(C1C(=C)C1)=O C1(NC(CC2(C)CCN2C(=O)CC2CNC(=O)O2)=O)C2CCCC1COC2 c1(CC(=O)NC2CC3(CN(C(CN(C(C)=O)C)=O)C3)C2)c(C)[nH]c2ccccc12 C(C(O)CC(=O)NCC1(O)CCCC1)NC(c1cc(CO)on1)=O N1(C(C(CSC)C)=O)CCC(c2nnc(CNC(C3(C)CC3)=O)s2)CC1 C(=O)(N=c1[nH]onc1C)C12C(CN(NC(=O)Nc3c(C)ccc(Cl)c3)C1)C2 c1(CC(=O)NC2CCN(C(C(CCC)=CCC)=O)C(C)C2)ccc([N+](=O)[O-])cc1 N1(C(c2cnc(CC)s2)=O)CC(NC(=O)CC(C)C2CCCO2)CC2(CCC2)C1 C1(OCC)CCCCN(C(c2cc(C)n(-c3ccc(Br)cc3)n2)=O)C1 C1(NC)CCN(Cc2ccccc2)CC1.C1(COc2ccccc2)C(=O)N1 Cc1c(C(=O)NC2CCC(CNC(=O)C(F)=C3CCC3)C2)sc2cncn12 c1(N2CCS(=O)CC2)[nH]c(=NCc2ccncc2)nc2sccc12 C1(CC(=O)N(CCCN(CC(=O)NCc2cccs2)C)C)CC(C)(C)CO1 C#Cc1ccc(C(=O)N(CCC(=O)NC2COCC2N=[N+]=[N-])C(C)C)cc1 c1(N(C(C)(C)C2CC2)C(N(C2C(C)CCCC2)CCO)=O)ccc2ccccc2n1 C(C(C)C)(C(O)C(=O)NC1CC2(C1)CC2C(=O)NC1CCOC12CCCC2)OC C1(NC(c2cc(OC)n[nH]2)=O)CC2CC(NC(=O)C(=Cc3cccs3)C)CC2C1 C1(C)(C(=O)Nc2c(OC)nn(C)c2)CC(O)CN1C(=O)COCC1CC1 C1(COC(C(CC)Oc2cccc(C)c2)=O)CCC2(CCCCCCC2)O1 c1(C(C)C(=O)NC2CCN(C(=O)CC(=O)N(C)C)C2C)ccc(CN(C)C)cc1 c1(C(=O)NC(CC)CNC(=O)CCCCCC#N)c(F)ccc2occc12 CCC(O)(CC)CCNC(=O)C1=CCC(NC(=O)C(C)N=[N+]=[N-])C1 c1(C(=O)NC2CN(C(C=C(C)C)=O)CC2Cc2ccccc2)c(Cl)c(C)nn1C c1(OC)ccc(-c2noc(C=Cc3cnc(C(=O)O)s3)n2)cn1 N1(C(C(C)NC(C)=O)=O)CCC(NC(c2cccc(C3CCC3)c2)=O)C1C C(C(C)CC(=O)NCC1CC2CC2N1C(=O)CCc1ccccc1C)OC C(=O)(C(C)S(N)(=O)=O)N(C1CCN(C(COCCC(C)C)=O)CC1)CCO c1(C(=O)NC)cn(CC(=O)N(C(C)CNC(=O)CCCn2cccn2)C)nn1 N1(C(c2nc(C)c(C)s2)=O)C2CC1CN(C(c1cnc[nH]1)=O)C2 C=C=CCC(=O)N(CCC(=O)NC(c1nncs1)C)C(C)C C1(C(=O)NCC2(F)CCN(C(c3cnn(CC)c3C)=O)C2)CN(C)CCN1C c1(OC)ccc(C(N2CC3CN(C(=O)Cc4ccc(F)cc4Br)C3C2)=O)c(Br)n1 c1(OC)ccc(C(=O)Nc2nccs2)cc1S(=O)(=O)Nc1cc2ncccn2n1 c1(C(N(C(c2ccc(OC)cc2)CC)CCO)=O)ccncc1N=[N+]=[N-] C1(CNC(CS(CC)=O)=O)CC(C(=O)N2CCC(C)(OC)CC2)=NO1 C1(C(=O)NCCNC(C(C(C)(C)C)SC)=O)CC1C1CCCCC1 CCCC(CC)CC(=O)NC1(CNC(C23CCC(CO)(CC2)CC3)=O)CC1 C1(C(=O)NC(C)CCN(C(=O)CN(C)C)C)COCCN1CC(F)F C1(NC(c2n(CC)cnn2)=O)CC(C)N(C(c2cccnc2F)=O)C1 c1(C(N(CCCN(C(=O)CCOC2CC2)C)C)=O)cc(Cl)c(Cl)n1C CC1CCCN(C(=O)C(C2CCCN(C(c3cccnn3)=O)C2)C)CC1 c1(-c2c(C)cc(OC(C)C)nc2)ccc2[nH]cc(CC(=O)Nc3cncs3)c2c1 n1(CC(=O)NCC(CNC(C(c2cnn(C)c2)OC)=O)F)nnc(=O)[nH]1 CC1C(NC(c2cnn(C)c2N)=O)CCCN1C(=O)Cc1ccn(C)c1 C(=O)(C(O)CCC(C)C)NCc1occ(C(=O)NC2(CC)CC2)c1 c1(C(=O)NC2C(NC(=O)C=Cc3nccs3)CCC2)ccc(O)c(Br)c1 C1(C(N(CC)CC2CCCO2)=O)CCCN1C(=O)CCOCCN(C)C CCC(C)C(O)C(=O)NC1CCC(NC(c2ccnn2C2CCC2)=O)CC1 C1(NC(c2ccnc(CO)c2)=O)COCCC1C(=O)NCc1ncco1 C1(OC)(CO)CN(C(=O)C(C2CCCO2)NC(C2CC2(Cl)Cl)=O)C1 C1(C(=O)Nc2nc(Br)cs2)CC(F)CN1Cc1cnc(-c2ccccc2)[nH]1 c1(OCC(=O)NC2C(NC(C3(C)CCCO3)=O)COC2)ccc(C(C)(C)C)cc1 c1(C(C(=O)NCC=C)N(C)CC2CCOCC2)ncn(C)n1 C(CC(C(=O)NCc1cc[nH]n1)NC(=O)C(F)CC1CCOC1)SC N1(C(=O)OC(C)(C)C)C(COC(c2cccc(Br)c2)=O)CCC2C1C2(F)F c1(N2CCC(C(CC)CC)C2)nc(=NCc2ncc(C)[nH]2)[nH]c2c(F)cccc12 C(=O)(CCC(C)(F)F)N1CCC(C2N(C(C3N(CC)CC3)=O)CC2(C)C)CC1 Cc1ncnc(C)c1C(N1CCC(NC(C2(C(=O)C3CC3)CC2)=O)C1)=O CC1CCCC(CC(=O)NC(C)CCCCNC(=O)Cc2cnn(C)c2)O1 N1(C(=O)CSC2CCCCO2)CC2CCCC(F)(F)C2C1 c1(O)cccc2cnn(C)c12.C1(CNC(=O)OC(C)(C)C)CC(C(=O)NC)CO1 N1(C(Cc2nc(C(C)C)on2)=O)CCOCC12CCN(C(=O)C(C)(C)C#N)C2 N1(C(C=CC=CCC)=O)CCOCCC1C(N1CCCC(CF)C1)=O N1(C(C(CC)N(CC)CC)=O)CCC(N(C(=O)C(C(C)C)n2cnnn2)C)CC1 N1(Cc2cn(CC(C)C)nc2)Cc2ccccc2CC1C(=O)NCc1cn[nH]c1 CCCC(C)(C)C(=O)N1CCC(C)C(CNC(C2(C#N)CCCCC2)=O)C1 C1(NC(CC2C(C)CCO2)=O)C2CC1CN(C(c1ccccc1F)=O)C2 C(C(C)(C)C(=O)NCC1CC(CNC(c2ccn(COC)n2)=O)C1)SC C1(NC(CNC(CC)=O)=O)CC(NC(c2cc(C)on2)=O)C12CCOCC2 N1(C(C2(SC)CC2)=O)CCC(c2ccccc2)(NC(=O)C=C2CCN(C)CC2)C1 C1CCCC2CC12.C1(CCNC(C(C)OC)=O)(NC(C2CC2)=O)CCCC1 C1(CNC(=O)C=Cc2ccoc2)CC2(CCN(C(=O)CCF)C2)CO1 N1(C(CNC(N)=O)=O)CC(NC(c2ccnc(CO)c2)=O)CC2(CC2)C1 c1(C(C(=O)NC2CC(C(C(=O)N(c3cnn(C)c3)CC)F)C2)C)ncc(C)s1 C1(CNC(C(CC2CC2)NC(C2C(C#N)C2)=O)=O)(CO)CC12CCC2 c1(C(=O)NC(CC(C)NC(=O)CC2CCN(C)C2=O)C)cnc2ccccc2n1 C1(C(=O)NC2CC(NC(=O)C=Cc3ccoc3)C2)CC(=O)C12CCC2 N1(C(C(C)C2CCCO2)=O)CCN(C(c2cn(C3CCC3)nn2)=O)CC1C1CC1 C1(NC(c2cc(C3(C)CC3)[nH]n2)=O)CN(C(=O)C#CC(C)(C)O)CC(F)(F)C1 N1(C(CSCC)=O)CC(=O)CC1C(=O)NCC(C1CC1)N(C)C c1(SCC)ccc(C(=O)NCC2(COC)CN(C(C3(F)CC3)=O)C2)c(F)c1F Cc1conc1CC(=O)N(CCC(=O)N(C)CCC1CCCN1C)C(C)C C1(NC(=O)CSCC2CCCO2)CC2CC(C1)CN(C(=O)C(C1CC1)C1CC1)C2 c1(C(N(C2CCN(C(c3cc(C(N)=O)[nH]n3)=O)C2)C)=O)cnc(S)nc1 C1(C(=O)NC(CNC(c2c(CC)ocn2)=O)CC(F)(F)F)CC12CCCCCC2 C1(C(=O)OC)(C(=O)NCC2CCN(C(=O)C3=C(Cl)CC3)C2)CC2(CCC2)C1 c1(C(N2CC=CC(NC(=O)C3=CCCCO3)C2)=O)oc2ccccc2c1CO C(C(O)C(=O)NCCN(C(=O)Cc1nocc1COC)C1CC1)=CC C1(O)(CN(C(C(C2CCCO2)OC)=O)C)CCN(C(c2cccnc2)=O)CC1 c1(CC(=O)NC2C(NC(COCC(=O)NC)=O)CC2)cnc2c(=O)[nH]ccn12 C1(C(=O)NCC(C)CNC(c2ccc(C(C)(F)F)cn2)=O)CCC(C2CC2)CC1 c1(C(=O)NC2CC(C)(NC(C=Cc3ccc(CC)o3)=O)C2)cc(Cl)ccc1F C=C(Br)CC(=O)NCCC1CC(NC(c2cc(C(F)(F)F)cs2)=O)C1 N1(C(Cn2ncc(C)c2)=O)CCN(C(C2(C)CC2Br)=O)CC1C c1(C(=O)OC(C(=O)OC)C2CC2)coc2cc(F)cc(F)c12 c1(CC)ccccc1C(N1CCC2CC12C(=O)NCC1CNC(=O)CO1)=O c1(C(N(C(C)CNC(C2CC2(F)F)=O)C)=O)cccc(-n2cccn2)c1 N1(C(c2ccc(CCCC)cc2)=O)CC(CNC(=O)C(C)C#N)C2(CC2)C1 CC(C)(C(=O)NC1CCN(C2CC2c2cccc(-c3cnsn3)c2)CC1)C(F)F C(CNC(=O)C(C1CCCOC1)OC)(C(C)C)NC(C1(CCCC)CCC1)=O c1(CC(=O)N(C(CCNC(c2ncn(CC)c2)=O)C)C)ccccc1C c1(CC)cccc(CC)c1NC(=O)CC1(NC(=O)CC2CCCCC2C)CCC1 N(C1CCCc2ccoc21)C(=O)NCc1c(F)cc(C)c(Br)n1 Cn1cnnc1CNC(=O)NC1CC1CNC(=O)OC(C)(C)C N1(C(C2CC(=C)C2)=O)CCC2CCN(C(=O)CN3CC4CCC3C4)CC12 N1(C(C(C)C2CC2)=O)CC2CCN(C(c3ccccc3Cl)=O)CC2C1 n1(Cc2ccc(C(N3CC(C=C)C(O)C3)=O)cc2)cc(Br)c(O)nc1=O N1(C(c2c(C(C)=O)coc2)=O)CCOCC(C)(CNC(=O)CN2CCCC2=O)C1 c1(CCNC(N(CC(O)C(F)(F)F)CCOC)=O)c(C)[nH]c2ccccc12 C1(CN(C)C(C2C3(CC3)C23CC3)=O)CCCN(C(=O)CC2(C)CCCS2)C1 C(=O)(C(C)(C=C)CCNC(C(C)OCCC=C)=O)NCC1(OC)CC1 N#Cc1ccc(=NCC(=O)N2CCC3(CC2)CC3NC(C2(CF)CC2)=O)[nH]c1 C(CN=c1ccc2cc(S(=O)(=O)NC34CC(C)(C3)C4)ccc2[nH]1)OCC(C)(C)C C1(NC(=O)CCc2cscn2)CCN(C(=O)C=Cc2cn[nH]c2)CC1F c1(CC(N2CCC(C(=O)NC(CCC)C3CC3)(C(C)C)C2)=O)cccc(O)c1F N1(CC(=O)NCC2CC(C)N(c3nc(C4CC4)ns3)C2)C(=O)NC(C)(C)C1=O N1(C(c2ncccc2Cl)=O)CC2(CCCCC2)CC1CO CC(C)(C(O)C(F)F)NC(c1ncoc1CNC(C1CC(O)C(F)C1)=O)=O CCC(CC(=O)N1CCN(C(c2cncc(O)c2)=O)C(C2CCC2)C1)CC(C)C c1(C(=O)NC(C(C)NC(CC(CC(C)C)C)=O)CO)cnc(O)c2ccccc12 C1(C(=O)NCCN(C(c2cnc(Cl)s2)=O)C(C)C)(CC)CC1(F)F c1(C(=O)NCC(CNC(c2cccnn2)=O)OC)cc(Cl)ccc1F C=CCCC(O)CN(C)C(C1(CNC(=O)COc2ccsc2)CC1)=O C(=O)(C(C)CCOC)N(C(C)CNC(=O)Cc1cccc(OC(C)=O)c1)CC C(=O)(C(CN(C)C)CC)N(CCN(C(C(C=C)O)=O)C)C(C)C c1(-c2ccc(CCCC)c(F)c2)n[nH]c2c1CCC(F)(F)C2 C1(C(=O)NC2CCN(C(C)=O)C2)CN(C(c2ccc(C(F)F)o2)=O)CC1(F)F C(=O)(CC1=CCOCC1)NC(CCC)C(=O)NCCC(C)(C)F C1(NC(CC(CCC)CC)=O)CC(O)(C2CCN(C(c3ccn(C)n3)=O)CC2)C1 c1(C(N2CCC(NC(=O)C=CC3CC3)C(CO)C2)=O)cc2c(cn1)COCC2 N1(C(C(C)=C2CCC2)=O)CCN(C(=O)C=Cc2ccc(C)s2)C2CCC12 n1(CC)ncc(C(N2CCC(CC(C)NC(C3(CO)CC3)=O)CC2)=O)c1Cl C(CN=c1[nH]c(N2CCOC(c3ccco3)C2)nc(=N)[nH]1)(C(C)(C)C)OC CCCC(C)(O)CC(=O)NCC(C1CCCC1)NC(=O)C(C)N(CC)CC C=CCCC(C1CC1)NC(=O)C(F)CC1CN(C(=O)CC2CC(F)C2)C1 c1(C(=O)NCC(CC=C)NC(=O)CNC(N)=O)cnc2cc(C)[nH]c2c1 C1(CC)CN(C(=O)C=C(C)CNC(C2(CO)CCCO2)=O)C(CC)CO1 N1(C(C(C)(C)OCC)=O)CC2C(CNC(=O)C(N3C(=O)CNC3=O)CC)C2C1 c1(C(N2CC(=O)NCC23CC3)C(=O)NC)cc2nc(Cl)ccc2s1 C(=O)(C(O)CCC(F)(F)F)N1CCOCC(NC(=O)CC2COCCO2)C1 N1(C(=O)OC(C)(C)C)CCC2CC(C1)CN(C(=O)C(c1cccc(Br)c1)NC)C2 C1(CNC(c2cnc(OCC)s2)=O)CCN(C(C2CCCCC2(F)F)=O)C(C)C1 Cc1ccc(C(=O)NCCC(C)(C)NC(=O)CCc2cnc[nH]2)cc1S(N)(=O)=O CC1CN(C(C2(CCO)CC2)=O)CC1CNC(c1cn(CCF)nn1)=O C12(CNC(C(C(C)C)SC)=O)CC(NC(=O)C(N3CCC(O)CC3)C)(C1)C(C)O2 c1(CCC(=O)NC2CC(CNC(CC=C=C)=O)C2(C)C)ccc(OC)c(F)c1 C1(CC)C(C(=O)NCCCCC2CN(C(C3CCO3)=O)C2)CCN1C c1(C(C)(C)C(=O)NC2CN(C(=O)Cn3cc(Cl)cn3)C2)ccccc1[N+](=O)[O-] c1(C(=O)NCCC(C)NC(C2(C3CCCO3)CCC2)=O)ccc(Cl)c([N+](=O)[O-])c1 c1(OC)ccc(C(C)(C)C2CC(=O)OCCNC(=O)N2)cc1Br.OC C1(C(N2CCCCC(NC(C(c3ccnn3C)C)=O)C2)=O)CCOC2(CCC2)C1 C1(CNC(=O)C=Cc2cncs2)CC2(CCOCC2)CN1C(=O)C(O)C(F)(F)F Cc1cccc(CC(N2CCCCC2CCN(C(=O)C(F)OC(F)(F)F)C)=O)c1 C(CCN=c1cc(C)nc(Cl)[nH]1)N(C(CC1CCCC(OC)C1)=O)CCO C1(NC(C2CCN2C(c2cnccn2)=O)=O)CCCCCC1O C12(NC(C3CC(C#N)C3)=O)CC(C1)N(C(c1cccc(N3CCCC3=O)c1)=O)C2 N1(C(c2cccnc2)=O)CCC2C(CCN2C(=O)CC2(O)CCOCC2)C1 C1(CCNC(CC2CC(=C)C2)=O)CCN(C(=O)C(C)CN(C)C)CC1(F)F C1(NC(C2(C)CC(F)(F)C2)=O)CCN(C(c2cccc(N)c2O)=O)CC1O CN1C(=O)CSC1CC(N1CC=CC1CNC(=O)CNC(c1ccccc1)=O)=O Cc1ccccc1C1(C(N2CC3C(C(=O)NCCN4CCS(=O)CC4)C3C2)=O)CC1 c1(OC)c(CN2CC3CN(C(=O)Nc4cccc(Cl)c4)CC23)cc(Cl)cc1Cl c1(C(=O)OCC)ccc(CC)c(N(C)C)c1.c12nncn1NC(=O)C2 N1(c2n(Cc3ccc(OC)nn3)nnn2)CC2CCN(C)CC2C1 c1(C(C)CC(=O)NCCN(C(=O)CCNC(=O)N(C)C)C)ccc(F)cc1F N1(C(COCCCC)=O)CCC(N(C(=O)Cc2cc(C)on2)C)C(C)C1 C(C1OCc2ccccc21)N(C(=O)Nc1cccc(S(=O)(=O)N(C)C(N)=O)c1)C C1(NC(COC(CNC(Cc2cc(C)[nH]n2)=O)(C)C)=O)CC(C)OC1=O c1(C(N(C2CCN(C(C3(CF)COC3)=O)C2)CCC)=O)cnn(C2CC2)c1 c1(C(=O)NCC(=C)CCNC(c2cc(C(=O)OC)n(C)n2)=O)ccc(C)nc1C CC1CCN(C(c2ccc(O)cc2)=O)CC1CC(N1CC(O)CC1CO)=O C(CCN=c1[nH]cc([N+](=O)[O-])cc1CO)NC(CC(CC)(C)C)=O C1(N(C)C(c2csc(-c3ccccn3)n2)=O)CCCCN(C(C2CCCO2)=O)C1 CC1(C)C(C(=O)NC2CCC(C)(NC(c3cccc(O)n3)=O)CC2)CCS1(=O)=O CC(C)C(C)C(CNC(=O)CCc1ccn(C)n1)NC(c1ccc(C#N)o1)=O C1(COC)(CNC(c2cncc(F)c2)=O)CCN(C(c2cc(C)c[nH]2)=O)C1 c1(C(=O)NC(CNC(C2ON=C(CC)C2)=O)(C)C)nc(Cl)cc(N)c1Cl N1(C(c2cccc(OCC)n2)CC)CCCC(C)CC1 C(=O)(CC1C(=O)Nc2c(Br)cccc21)N1C(COCC)CCCC1 c1(-c2scc(C(N3CCOCC3)=O)n2)c(F)ccc(O)c1F S(=O)(=O)(c1ccc2c(c1)CCC(=O)N2)Nc1cc(N)c(OCc2ccco2)cc1 C1(C(=O)O)CC2(CCN(C(=O)C=CC(C3CCCCC3)=O)CC2)C1 Cc1nc(Cl)cc(=NCC(C)(C2CC2)NC(=O)CC2CCC(C(F)(F)F)O2)[nH]1 N1(C(C(CC)F)=O)CCC(NC(=O)CN2CCCS2(=O)=O)C(CC)C1 C(=O)(C1=NOCC1)NCC(CC)NC(=O)CC1(N(C)C)CCC1 N1(C(CCOc2c(CC)cccc2)=O)CC2(CCC2NC(C2(SC)CC2)=O)C1 c12cccc(c1NC(=O)CSC(F)F)SC2.c1(C(=O)OC)ccc(CN)cc1 C(=O)(C1=C(c2ccccc2)SCCO1)N1CCC(NC(CC(C)OC)=O)CC1 N1(C(C=C2CCC(C)C2)=O)CCOC2(C1)CN(C(C1CC3(CCCC3)CO1)=O)C2 C=C(C)C1CN(C(=O)C(C)CNC(=O)CCCC(C)C)CCO1 c1(NCCC(CCC)C)nc(N(CC(C)OC)C)nc2c1ncn2CC C(=O)(C(F)(F)CC(=O)NC(C)CCc1ccccc1)OCC CC(CC(=O)N1CC(O)C2(CCC2)C1)C(C)(C)NC(C1CC12CC2)=O C12(C(N3CCC(CC#C)C3)=O)CC1CN(C(=O)Cc1csc(C)n1)C2 c1(C(C)C)ccc(C(C)NC(c2ccc(OC(F)(F)Cl)cc2)=O)cc1 C(C1=CN(C(=O)OC(C)(C)C)CCC1)(n1ccnc1C(O)CC)OCCC N1(C(CCSC)=O)CCCC(CN(C(=O)CCCOC(C)=O)C)C1 C(CC)(C(=O)NCC1(NC(C2CCN(C(C)=O)C2)=O)CC1)OCC C1(C)(CC)CCCN(C(=O)CC(C2CC2)NC(=O)C(C)n2cccc2)C1 N1(C(C)=O)CCCCC1C(=O)NCC1COCC1NC(C1(C)CCCC1)=O CC(O)C(C)(C)C(=O)NCC1(O)CN(C(c2cccc(C(N)=O)c2F)=O)C1 S(=O)(=O)(C1CCCN(C(C)(C)C)C1)NC(c1nn(C(CC)C)c(C)c1)=O c1(CC)cc(N2CCC(CNC(C3CC3F)=O)C2(C)C)nc(C)n1 C1(CN(CCOC)Cc2ccccc2)CCCN1c1nc(C)ns1 C1(CNC(C(COC)(C)C)=O)CCCCCN1C(c1cccc(F)c1F)=O c1(C(N(C(C)C)C)=O)cc(CNC(=O)C=Cc2cc[nH]c2)[nH]n1 CCC(CC(C)C)C(=O)NCC12CC(C1)C(NC(c1cnoc1C)=O)CO2 N1(C(CCCCOCCC=C)=O)CC(C2(NC(c3nc(C)n(C)c3C)=O)CC2)C1 N1(C(=O)OC)CCCC(C(=O)Nc2cc(C(F)(F)F)ccc2N2CCCC2)C1C c1(C(N2CC(COC)(CNC(c3nc(C)oc3OC)=O)C2)=O)cc([N+](=O)[O-])n[nH]1 N1(C(COCCN(C)C)=O)CCN(C)CC1CNC(C1CC(O)CC(=O)N1)=O C=C(C)CCC(=O)NCC(C1CCC1)NC(=O)C(C(C)C)c1ccc(Cl)cc1 CC(C)CC(C(=O)NC1COCC1O)N(C)C(c1cccc[n+]1[O-])=O C(C(=O)NC1(C(=O)NCc2ccc(C)cn2)CC(F)C1)(C(C)(C)C)OC C1(CC(=O)NC2(CF)CN(C(c3cnns3)=O)C2)CCCCC1(F)F C1(F)(N(C(=O)OC(C)C)Cc2ccc(=O)n(C)c2)CCCCCC1 S(=O)(=O)(c1cnc(C(F)(F)F)c(F)c1)N(C1C(SC)CCCC1)C c1(C(=O)NCCN(C(=O)CC2CCC(C(C)C)O2)CC)cc(C)oc1C(F)(F)F C(=O)(CC(C(F)F)NC(=O)C(C1CCCCC1)=O)NCc1nc(CC)oc1 Cc1nc(O)ccc1C(=O)NC(CC1CCOCC1)C(=O)NCC1(C)CCCO1 C(=O)(C(C)(C)OCC(F)(F)F)NC(C)C(C)NC(c1csc(-c2ccsc2)n1)=O C1(C(=O)NCCN(CCC)CCC)CCCCCCN1C(=O)C(C)n1cccn1 C1(C)(OCC(=O)N(CC(C)CNC(=O)C=CCO)C)CCOCC1 C1(NC(=O)CC2CCCCC2NC(C2C3CCC(F)C23)=O)CCC2(CCC2)C1 CC1CN(C(=O)CC2COCCOC2)CCC1C(N1CCC(O)(C(=O)N(C)C)C1)=O C(C(C(C)C(C)C)NC(=O)COc1ccsn1)NC(Cc1nc(C)[nH]n1)=O Cc1cc(C)c(C(N2CC(N(C(=O)CCOCC(C)C)C)C(O)C2)=O)cn1 C(=O)(C(C)C(F)(F)F)NC1CC(C(C)NC(CCC(=O)NCCC)=O)C1 CCCCCCCCC(F)C(=O)NCCOC1CCN(C(=O)C=CC2CCC2)CC1 Cc1conc1C(=O)N(C1(C(N2CCCC2C2(C)CC2)=O)CC1)C C1(C(=O)NCC(C)(C)O)CCN(C(C23CC(F)(C2)C3)=O)CC1 C1(C)(C(=O)NCCCC(C)NC(c2c(C)c[nH]c2CC(N)=O)=O)CCC(F)(F)C1 c1(C(=O)NCC(C)(C)CNC(C2CCC(F)C2)=O)cccc2nc(S)oc12 CC1=NOC(C)(C(=O)NCC2CCN(C(=O)Cc3cncc(Br)c3)C2)C1 CN1CCC(C(=O)NCC2(Cl)CC2(F)F)S1(=O)=O c1(C(=O)NC2CN(C(CC(CC)SC)=O)CC2O)ccc(SC)cc1Cl c1(NC2CC(S(C)(=O)=O)C2)nccc(=NCc2nc(O)n[nH]2)[nH]1 c1(NC2C(C(=O)NCC(=O)NC34CCC(C3)C4)COC2)ccc(O)cc1 Cn1ncc(C#N)c1N(CCN)CC1CC2CC2N1C(=O)C=Cc1ccccc1 C(=O)(C(C#N)C(C)(C)C)N1C(C)CCC(NC(c2c(C(C)C)nns2)=O)C1 c1(C(=O)NC(C)CN(C)C(C2CCCC2(C)C)=O)cccc(=S)n1O N1(C(C(C)SCCCC)=O)CCC(O)(CN(C)C(c2nccn2CC)=O)C1 N1(C(C(C2CCC2)OCC)=O)CCC(O)(CCNC(=O)CSC)C1 C1(N(C(=O)COCCNC(C2C=CCCC2)=O)C)CCCC1C#N c1(C(N2CC(CNC(c3ccnc(Cl)c3Cl)=O)OCC2)=O)cccc(F)c1F N1(C(CCc2ccc(=N)[nH]c2)=O)CCCC2CN(C(c3cccs3)=O)CC12 N1(C(C2CC(C(C)(C)C)C2)=O)CCC2(CC1)CC2CN(C)Cc1cccnc1N CC1=C(C(=O)NN2CCCC2C(=O)NC23CCC(C2)OC3C)CCCO1 CC#CCC(C(=O)N(CCO)CCO)NC(C1C2CCC(F)C12)=O c1(C(C(=O)NCCCC)N(C)Cc2ncc[nH]2)cc2sc(C(=O)OC)cc2o1 c1(-c2ccc(NCc3cc(C)nn3C)c(F)c2)csc2ccccc12 C=CCCC(Cc1ccccc1)NCC(c1ccsc1)C N1(C(C2(C)CCN(C(C(CC=CCC)C)=O)C2)=O)CCN2CC(O)CC2C1 N1(CC(C)C)CCN(C(=O)C(=O)NCC(C)Cn2cccn2)C(C)C1=O c1(C(=O)NC2CCCC(NC(C(C)C)=O)C2)cc2ccncc2s1 N1(CC(=O)NC2(C)CC(NC(c3c(C)onc3CO)=O)C2)CCS(=O)(=O)CC1 C(=O)(CCCCO)NC(C1CN(C(=O)CN2CCOCC2)C1)C C#CCS(=O)(=O)CCNC(=NCCSC1CCCC1)NC1CCN(C(=O)OC)C1 Cc1cccc2c1OCC2C(=O)N(C(C)CN(C)C(c1cnc(O)n1C)=O)C c1(C(=O)NCC2CC(NC(c3ccc(Cl)cn3)=O)C2)nc(Cl)ccc1Cl N(C(=NCC1(C(=O)OC(C)(C)C)CCC1)NCC12CC(CO1)C2)C(C=C)C c1(C(N(CCCNC(c2ncnn2C)=O)CCC)=O)n[nH]c2c1COC2 C(=O)(CCCN1CCCC1)N(C(CCNC(COCCCCOC(C)=O)=O)C)C c1(CNC(c2c(C)onc2)=O)cccc(NC(=O)CCN2CCC(F)C2)c1 N1(C(c2c(N)non2)=O)CC2COCC(C1)C2NC(=O)Cc1cnns1 C1(CC(=O)NCCNC(=O)NCC)CCCN(C(C2CCC(=O)NC2)=O)CC1 N1(C(C(CC)OC)=O)CCN(C(c2n[nH]c(C)c2F)=O)C(C(C)C)C1 C(c1cccnc1)=CC(=O)NC1CC(NC(C(C)Cc2ccncc2)=O)C1 CC1(C)CC(C(=O)NC2(CCCNC(=O)C(CC(F)F)C3CCC3)CC2)=NO1 c1(C(=O)NCCCN(C(=O)C(c2cccnc2)O)CC)cccc2[nH]ncc12 c1(NCC(CCCC)NC(=O)CC(CN(C)C)CC)ncnn2c(Br)ccc12 CCC(CC(=O)NCCC1(NC(=O)C(C)Cc2ccncc2)CC1)SC c1(C(N(C2CCCN(C(CC(C=C)CC)=O)C2)CCF)=O)ccc(F)c(C)c1Cl c1(C(=O)NCC2(C)CCN(C(C3CCCN3C3CC3)=O)C2)cccn2nnnc12 Cc1ccc(C(=O)NC2(C)CCN(C(C3CC34CC(O)C4)=O)C2)nc1 Cc1cc(F)cc(C(=O)NC2CC(NC(=O)C(F)(F)c3ccccn3)C2)c1N c1(C(N(CC(C)NC(C2CC(OC(C)(C)C)C2)=O)C)=O)cc([N+](=O)[O-])ccc1Cl c1(C(N2CCC(CNC(C3(O)CCOCC3)=O)C2)=O)cc2cccn2cn1 CCCCC(C(=O)N1CC(S(N)(=O)=O)C1)NC(c1cnn(C(C)C)c1)=O c1(NC(=O)NC2CCC(OC)C2)cccc(N2CCN(C)CC2)c1C CC1(C)CC1(C#N)C(N1CCC(CNC(=O)CCNC(C2CCC2)=O)C1)=O N1(C(=O)C2=CCCN(Cc3cc[nH]n3)C2)CCc2[nH]c3ccccc3c2C1 C(C(C)(C(=O)N1CCCCC1)NC(=O)NCc1cnc(N(C)C)o1)OC C1(c2nn(C(C)C(F)(F)F)c(-c3cnc(O)s3)n2)CCOC2(CCOCC2)C1 C1(C)(OC)CCCN(C(=O)C(C)(C)C2CCCN2C(=O)CSCCC(C)C)CC1 n1(CC)nnc2c1C(C(=O)NC1CCCC1)CN(C(c1nc[nH]n1)=O)C2 C(N=c1[nH]c(=NCC2(C)CCC(=O)N2)c2ccccc2[nH]1)C1(C)CCCCC1 c1(CSC)ccc(C(=O)NCC2(CNC(C3CN(C)CC3C)=O)CC2)cc1 N1(C(c2cncc(C)c2)=O)CC2CCC2(CNC(=O)C(C)CC(C)C)C1 C=CCC(CC)C(=O)NC1CC(C(=O)NCCN2CCC(C)(C)C2)CC1O CCC(C)C(=O)NCC(=O)N(CC(O)CNC(c1cn(C2CC2)nn1)=O)C c1(NC(c2ncccc2NC(c2csnn2)=O)=O)cc2cc(F)ccc2cn1 N1(C(C2N(C(c3ccc(C(N)=O)nc3)=O)CC(O)C2)=O)Cc2ccc(O)cc2C1 N1(C(c2c(CC)nnc(C)c2)=O)CC2CC3CC2C1C3NC(=O)C#CC(C)C c1(C(=O)NCC(C)N(C)C(c2cc(CO)on2)=O)cnc(N)cn1 C(=O)(C1=CC(C)(C)C1)NCC1(O)CC(CNC(CCc2n(C)ncc2)=O)C1 C(=O)(C(CC(C)(C)C)OC)NC(C(=O)N(C)Cc1n(CC)ncc1)CN(C)C C#CC1CCN(C(=O)CCC2CCN(C(C3(CO)CCC3)=O)CC2)C1 N1(C(c2scc(COC)c2)=O)CCC2(CC(NC(=O)C(C)(C)F)CO2)C1 CC1CCN(CC(=O)NCc2occc2C(=O)NC2COCC2C)CC1 C(CC(C(=O)NC1(CC(N2CC(O)(CO)C2)=O)CCCCC1)OC)OC c1(C(N2CCC(NC(=O)Cc3nnc(O)s3)(CO)C2)=O)cc(F)c(CO)c(F)c1 C1(CCC)CCC(c2nnnn2CC)(NC(c2cccc(F)c2)CF)CC1 N1(CCC(N2CC3C(CNC(C4(CC)CCC4)=O)C3C2)=O)C(=O)NC(C)(C)C1=O C1(CNC(c2coc(O)n2)=O)CC12CCN(C(c1c(Cl)nsc1Cl)=O)CC2 C(=O)(C1=C(C)C(C)(C)OC1=O)N1CCC(COC)(NC(c2cnc(Cl)s2)=O)CC1 c1(NC(c2c(CC)nccc2)=O)ccc(Br)c(C)c1C.N12CCN(CC1)CC2=O c1(C(N2CC(C)OCC2C)C(=O)NCCCSCC)cc2ccccc2nc1C N1(C(c2[nH]cc(CC)n2)=O)CCN(C(=O)C(O)CN(C)C)CC12CCC2 N1(C(CCC2(NC(C(C3CC3)OCC)=O)CCCC2)=O)CCC(C2CCOC2)C1 C1(C(=O)NCCNC(C2(C)CC2)=O)CCCN(C(C2(CO)CC2)=O)C1 C1(CN(C(CCCOC(C)C)=O)C)COCCN1C(=O)C(O)C1CCCC1 C1(NC(C2(COC)CC=CC2)=O)CC2(C1)CN(C(c1cc(C(N)=O)cn1C)=O)C2 N1(C(COCCCCCC)=O)CCC(COC)(NC(=O)C(c2cccnc2)O)C1 C1(N(C(CCCN(C)C)=O)C)CCCN(C(C2(P(C)(C)=O)CC2)=O)CC1 C12(CNCC(C)C3CCC3)CCC(C(=O)O)(CC1)OC2 C(CC(O)CNC(=O)CCc1nc(C)no1)NC(C=C(C)Cl)=O N1(C(C(CC)N(C)C)=O)CCN(C(c2cc(Br)c(F)cc2C)=O)CC(O)C1 N1(S(CCOC)(=O)=O)CC2(CCC(NC(c3ncc(Br)cc3F)=O)CC2)C1 c1(CC)nnsc1C(=O)NC1COCC1C(=O)NCCC1(C)CCCO1 c1(C(N2CC(CNC(=O)C(=Cc3c[nH]cn3)F)C2)=O)cnc2ncc(Cl)cn12 CCCCC(O)C(=O)N(C1CCCCCC1)CCNC(=O)CN1CC(CC)C1 Cc1ccc(C(=O)NCC(CC2CC2)C(=O)N2CC(N3CC(F)C3)C2)c(C)c1 C1(F)(C(=O)NCC(CC)NC(=O)C(C)(C)N2CCOCC2)CCC(C)CC1 CC1CN(C(c2ccc(N(C)C)cn2)=O)CC1NC(C1CCCC1CF)=O c1(CN2C(CC(=O)NC(c3ccno3)C)COCC2)csc2ccccc12 C(C1CCN(C(=O)C(C)C2CC2)CC1)=CC(N1C(CCC=C)CCC1)=O N1(C(COCCCCCC)=O)CC2CCOCC2(NC(c2ccc(=N)[nH]n2)=O)C1 c1(CC(=O)NC(C(=O)NC(C=C)CO)C)cn(C)cn1 c1(NC2CCN(S(CC)(=O)=O)C2)ccc(S(=O)(=O)NCC2(CC#N)CC2)cc1Br S(=O)(=O)(c1ccc(I)cc1)N1C(C(=O)Nc2cnc(C)nc2C)CC(O)C1 CC1CCCCN1CCCNC(N1CCC(C(C2(n3cccc3)CC2)=O)CC1)=O C1(C(C)CC(=O)O)CCN(C(c2nscc2Br)=O)CC1 c1(N2CC(C)(C)C(NC(=O)C=Cc3ccco3)CC2)ncnc2cccc(F)c12 n1(C(C)C)cc2c(n1)CC(NC(N1CCCC(c3ccon3)C1)=O)CC2 N1(C(C(=O)NCC2C(C)CCO2)=O)CCN(CC(=O)NC2CCC2)CC1 C(=O)(C(F)(F)C(O)C(C)C)NC(C1OCCN(C(C(C)OC)=O)C1)C C(=O)(C(C)S(=O)(=O)C(C)C)NCCCN(C(c1cc(N)c(C)cc1C)=O)CC N1(C(c2c(SC)ccs2)=O)CCC2C(C1)CN2C(c1conc1C)=O C(=O)(C(C)CC(N)=O)NCC(c1c(OC)cccc1)NC(=O)C1=NOCC1 N1(C(C(CC#C)O)=O)CC2CC(C(=O)NC(c3ccccc3)CC=C)CC2C1 Cc1cc(F)ccc1C(=O)NC1CCCC(CNC(C2CCS2(=O)=O)=O)C1 CC(CCCCNC(=O)CC1CCC(=O)N1C)NC(=O)CNC(=O)CC(F)(F)F C=C(CNC(=O)COCCNC(=O)C(F)C1CCOC1)CC C(=O)(C(C)CC(=O)c1ccc(F)cc1)NCC(CNC(c1cnc(O)s1)=O)OC Cc1cc(C2CCCN2CCCC2CCOC2)cs1 N1(C(CCC(CC)OC)=O)CC2=C(C1)CN(C(=O)C(C)Sc1ncccn1)C2 CC(C)CC(CNC(C1NC(=O)OC1(C)C)=O)C(=O)N(C)CC1COCCO1 N1(C(C(C)=CC)=O)CCOC(CCNC(=O)CC2(O)CCCOC2)C1 c1(C(=O)NCC(CCNC(C2CC(Cl)(Cl)C2)=O)OC)cn2c(C)cccc2n1 N1(C(c2c(C(=O)OC)cco2)=O)CCCC(NC(C2CC(C(C)C)=NO2)=O)CC1 c1(C2C(NC(C(C)(C)C3(C)CC3(F)F)=O)CCC2)cc(Cl)cc(Cl)c1 c1(CC)nc(C)c(CNC2(c3ncc(C)o3)CC2)o1 C=C(C)C1OCCCC1C(=O)NCC(C)(C1CC1)NC(=O)Cn1ncnn1 C1(C(=O)Nc2cccc(C)n2)CNC(=O)C12CCN(C(=O)CCC(C)C)CC2 C1(C(N(C)CCNC(c2ccoc2)=O)=O)C2CCC1(c1ccc(F)cc1)C2 C1(C(N2C(CCNC(c3nc(OC)c(C)s3)=O)CCCC2)=O)C2CC(F)(F)CC12 c1(C(=O)NCC(CC)NC(=O)C(C)n2cncn2)c(Cl)cccc1[N+](=O)[O-] C(C(O)C(=O)NCC(C)N(C)CCC)NC(CSCCC)=O C1(C(=O)NCCC(=O)NCC(C)(O)C2(C)CC2)(OC)CCSC1 c1(C(=O)NCCOCCN(C)C(c2c(N)cccc2Cl)=O)nccc(Cl)c1F C12(CNC(C(C)SC)=O)CC(CO1)N(C(=O)C(C)COc1ccccc1)C2 CN1CCC(CC(N2CCC(O)C2C(=O)NC(C2CCCCC2)CO)=O)CC1 C1(OCCOC)CCN(C(c2cccc(OC)n2)=O)CC1.c12n[nH]cc1NC2=O N12CCN(CC1)CCCNC(=O)C1(COC1)C2=O.C1(CC)CCC(N(C)C)CC1 C1(NC(C(CC=C)CNC(=O)CSc2cn[nH]c2)=O)CCn2cncc2C1 N1(C(CS(=O)(=O)NC)=O)CC(CNC(C2CCC(O)CC2)=O)C(C)(C)C1 C1(C(N(C(CN(C(c2c(OC)csc2)=O)C)C)C)=O)CCc2cnnn2C1 c1(C(=O)NC(C2(O)CN(C(=O)CC3(C)CC(F)(F)C3)C2)C)cc(F)cc2nn[nH]c12 N1(C(c2cc(C(C)(C)C)no2)=O)CCC(NC(C2(C)CC=CCC2)=O)C(C)(C)C1 CC1(C)CCCC(CC(N2CCN(C(=O)C3=COCCO3)C(CCO)C2)=O)C1 CS(=O)(=O)C1CCCC1C(=O)NCC1CCN(C(c2cc(CO)on2)=O)C1 c1(NC(c2c(C)scc2)=O)cccc(NC(=O)C=Cc2cn[nH]c2)c1 c1(C(N2CCC3(CCCN3C(=O)C(O)C(F)(F)F)C2)=O)cc2cc(Cl)cnc2o1 CC1(C(=O)NCC2CCN(C(C3CCC(=O)C3)=O)CC2)CCNC(=O)C1 C1(NC(CCN(C)CC)=O)CC2CCC1CN(C(=O)C(c1ccc(C)s1)C)C2 c1(C(C(=O)N(CC(C)CNC(=O)CC2CCC2)C)(F)F)ccc(Cl)cn1 N1(S(CC=C)(=O)=O)CCC2CC(C(N3CCC4(C3)CN(C)C4)=O)C2C1 Cc1ccc(C(N)=O)cc1C(=O)NCC(C)(C)NC(=O)Cn1cn[nH]c1=N Cc1ccc(S(N)(=O)=O)cc1C(=O)NC1CC(C)CN(C(c2nonc2N)=O)C1 N1(C(C(C(=C)C)(C)C)=O)CCN(C(C2CCCC2S(C)(=O)=O)=O)CC(C)(C)C1 CC1(C)CC1(c1cccs1)C(=O)NCC1CCN1C(=O)CNC(c1cscn1)=O C1(NC(C2CCCC23CC3)=O)CC2CCC1N2C(=O)Cc1ccccc1 O=C(NNC(=O)c1ccc(-c2nncn2C2CC2)cc1)NC1CCCCO1 C1(NC(C2CCOC2=O)=O)CCCCN(C(=O)Cn2cc(C(F)(F)F)cn2)C1 Cc1cc(C(=O)NCC2CCN2C(=O)C(c2ccccc2)C2CC2)c(F)c(Br)c1 NC(=O)CC(O)CC(=O)N(CCNC(=O)C(F)(F)C(F)F)Cc1ccccc1 c1(OC)ccc2ccnc(C(C)NC3CC4CC3C3CCCC43)c2c1 C1(C(C)NC(c2ccc(F)cc2)=O)CN(C(=O)CCCc2nncn2C)CCO1 c1(C(=O)NCC2(F)CCC(CNC(CC(C)(F)F)=O)CC2)cc2ccncc2[nH]1 Cc1ncc2n1CC(C(N1CCC(C(C)Nc3ncnc(=N)[nH]3)CC1)=O)CC2 C1(C(=O)NC(C(C)C)CCNC(C2(F)CCC2)=O)CCC(C)(F)CC1 n1(CC(=O)NC2CCCN(C(c3cccnc3Cl)=O)CC2)nc(Cl)ccc1=O C(=O)(C(F)CC(C)(C)C)c1cn(C)nc1.N1CC(F)(F)C1(C)C CC1(C#CC(=O)NCC2CCN(C(=O)C(C3CCCO3)C3CC3)C2)CC1 c1(OC)ccc(C(=O)NC(C)CN(C(=O)C(CC2CC2)OC)C)nc1Br C(=O)(C(F)=C1CCCC1)N(C(CNC(CSCC=C)=O)C)CC c1(N(CCO)CC2(C)CCC2)nnc(-c2cnccn2)n1Cc1ccsc1 N1(C(C2(C)CN(C)C(=O)CC2)=O)CC2(C1)C(NC(=O)CCC(N)=O)CCS2(=O)=O N1(C(c2c(C#N)ccs2)=O)CCC2CN(C(c3ccc4ncnn4c3)=O)CCC12 C(=O)(C1(C)CCc2cc(C)ccc21)N1C(OC(N(CC)CC)=O)CCCC1 C1(CNC(C2CS(=O)(=O)C2)=O)CN(C(=O)Cc2cscn2)CCO1 Cc1cc(C(=O)NCCNC(C2C3CCC2(c2cscn2)C3)=O)cc(C)c1 C1(C(N(C(C)CCNC(=O)CCc2ccc(O)cc2)C)=O)CS(=O)(=O)CC12CC2 c1(C(=O)NC(C(C(C)C)NC(=O)CCc2cnn[nH]2)C)cnnc2ccccc12 CCC(C)(CNC(c1sccc1CO)=O)NC(=O)Cc1cccnc1 C(=O)(C1=COc2ccccc2O1)NC1CN(C(C(C)SCC)=O)C2(C1)CCC2 C1(C(=O)NCC2CC(NC(c3n(C)c(S)nn3)=O)C2)CCC(C)(C)CC1 C(=O)(CC(C)C(C)(C)C)NC(CC1CN(C(c2nn(CC)nc2C)=O)C1)C Cc1cc(C(F)(F)F)nn1CC(=O)NCCC(C(C)C)NC(C1CC12CCC2)=O C(=O)(C(C)CC(C)(F)F)NC1(C)CCN(C(c2ccc(OC)nc2C)=O)C1 CCCC(CCC)=CC(=O)NCC1CN(C(C2CCCC2)=O)CC1C c1(C(N2C(C(=O)NCc3c(C(=O)OC)[nH]cc3)CC2C)=O)ccnc(CO)c1 C(C(=O)NCC1COCC1NC(=O)CCc1cnco1)(C(C)C)OC Cc1cc(C(=O)N(C(C)CN(C(=O)CC2CCCC2O)C)C)ccc1S(N)(=O)=O N(C(=NCCN(c1ccccc1F)C)NCCNC1CCC1)CC(NOC)=O c1(C(N2CCC2CNC(=O)C(O)C2CC2)=O)ccc(NC2CC=CCC2)cc1 c1(C(N(CCCCNC(c2cc(COC)no2)=O)C)=O)cncc(CO)c1 CC1CN(C(=O)CSc2ccccn2)CC1NC(c1csnc1Cl)=O C#CC1(O)CCCN(C(=O)C(CN(C(=O)CCc2cn(C)nn2)CC)N(C)C)C1 c1(C(N2CCN(C(C(c3scc(C)n3)C)=O)CC2CO)=O)cn(C)c(=O)cc1C c1(SCCNC(N(C(COC)CC2CCCC2)C)=O)ccccc1F CC1CC(C)(C)N1C(=O)CC1CCN(C(=O)CCOC2CCC2)CC1 C1(CCC(=O)NC2CN(C(c3cn(C4COC4)nn3)=O)CC2O)NC(=O)NC1=O N1(C(CSCC)=O)CCN(C(=O)C(C(C)C)N(C)C)CC(O)C1 Cc1ccccc1C(CC(=O)OC(C)C)NC(N1CCOC(CC(F)(F)F)C1)=O N1(C(=O)CCC2OCCO2)CCCC2(CCN(C(=O)CN3C(=O)CCC3=O)C2)C1 c1(OCC(C)C)ccccc1C(N1CC(n2cc(CC(=O)O)nn2)C(C)C1)=O c1(CN2CCC(O)(C(N3CC4C(C3)C4(F)F)=O)C2)c(O)cc(O)cc1O C1(CC=C)(NC(=O)CC2COCCO2)CCN(C(c2cccn2C)=O)C1 C1(C(C(=O)NCCC)N(C(C)C)Cc2ccncc2)CCCC(CC)C1 c1(C(N2CC=CC(NC(COC(CC)(C)C)=O)C2)=O)c(C)nn2ccccc12 C(c1cncc(C)c1)=CC(=O)NC1(CC=C)CN(C(C2(C)CS(=O)(=O)C2)=O)C1 c1(NC(C(N2CCC(N(C(c3nc(C)n(C)n3)=O)C)C2)=O)C)ccc(Cl)cc1Cl C12(NC(C=C(C)Cl)=O)CCC(CC1)N(C(=O)C(C)CC(C)C)C2 c1(CC(=O)NCCC(C)N(C)C(c2ccnc(O)c2)=O)cc(F)cc(F)c1 Cc1ccc(F)c2oc(C(=O)NC(C)CN(C(=O)COc3cccnc3)C)cc12 c1(C(C(N2CC(C)CC(NC(COCC)=O)C2)=O)(C)O)cccc2ccccc12 CC(CF)CC(=O)N1CC2C(NC(c3cnc(-n4cccn4)cn3)=O)C2C1 C1(N(CC#C)C(C2CC(C)=NO2)=O)CCN(C(=O)CCC=CC(C)C)CC1 C1(Nc2ccc(C(=O)OC)cn2)CN(C(=O)CC2COC(=O)C2)CC1(C)C C1(Cc2ncc(C(=O)OC)s2)CCN(C(=O)CN2CC(CN(C)C)C2)CC1 N1(C(c2cccc(SC)c2)=O)CCC2(CCC(NC(=O)CC3(O)CCC3)C2)C1 N1(C(c2c(C)occ2)=O)CC(NC(C2COC(C)(C)CO2)=O)C2(CC2)C1 C1(NC(C2(C(N)=O)CC2)=O)CC2CC(C1)CN(C(c1ccc(Br)o1)=O)C2 c1(NC(C2CCCN(Cc3c(C)n(C)nc3)CC2)=O)c(O)cccc1C#N CC1CCN(C(c2nn[nH]c2Cl)=O)CCN1C(=O)Cc1cccc2nsnc12 c1(C(N(C2CC(NC(c3c[nH]nc3F)=O)C2)C)=O)ccc(F)cc1Cl CC1CCC(NC(C2(C)CCCO2)=O)CN1C(C1CCC(C(F)(F)F)CC1)=O CCC(C)(C)C(C)CC(=O)N1CCC(C)(NC(=O)C(c2c(C)noc2C)C)CC1 c1(NC(c2c(CNC(C(CC)COC)=O)cc[nH]2)=O)cc(C)cc(O)c1 C1(COC)(NC(=O)CC(C)CF)CCCN(C(C2(COC)CC=CC2)=O)C1 Cc1c(F)ccc(CN2CC(C)CC2C(=O)NCc2cnn(C)c2)c1Cl c1(-c2cn(CCN(C(=O)C(F)(F)C3CCCC3)CC)nn2)cccc(N)n1 Cc1c(Cl)cnn1CC(=O)NCC1CN(C(C2CC2c2cccnc2)=O)CC1O c1(CC(=O)N(CC(C)(C)CNC(C2CCCS2)=O)C)ccc2ccoc2c1 C1(O)(C(N(CC(CN(C(CC2CC(=C)C2)=O)C)O)C)=O)CCCCCC1 Cc1ccncc1C=CC(=O)NCC1(F)CCCN(c2nnc(CO)s2)C1 C1(CC=C)(NC(C2(C(F)F)CC2(F)F)=O)CN(C(c2csc(NC(C)=O)n2)=O)C1 C(=O)(C1=CC2CCCCC12)N1CC2N(C(CCCC(C)C)=O)CC(C2)C1 N1(CC(=O)NCC2C(NC(C(N3CCN(C)CC3)C)=O)C2)CCC(C)(O)C1 C=CCC(CC=C)C(=O)NC(C)CC1CN(C(=O)C(C2(O)CCCC2)F)C1 C1(CC(=O)N(C)CC2CN(C(=O)Cc3nc[nH]n3)C2)COC(C)(C)CO1 N1(C(CCOCC#C)=O)CCC2CN(C(C3(N(C)C)CCOCC3)=O)CC12 N1(C(C2(CCC=C)CC2)=O)CC2CCN(C(c3ccc4nc[nH]c4n3)=O)CC2C1 c1(OC)ncccc1C(N1CCC(N(C(=O)COc2ccsc2)CCO)C1)=O C1(C(N2CCC(NC(c3cc(C(N)=O)no3)=O)(CF)C2)=O)CCCC2C1C2(F)F C12(CNC(c3ccc(C)cc3)=O)CCC(CC1)N(C(=O)CC(O)CC(C)C)C2 c1(CC(N2CCC(N(C)Oc3c(CC)cccn3)C2)=O)cn2c(C)csc2n1 C1(C(=O)Nc2ccc(C)nc2)CN(Cc2ncn(C)n2)CCC1(F)F c1(C(=O)OC)ccc(COC2CC(CNC(=O)OC(C)(C)C)C2)cc1 C1(CN(C(c2ncsc2C)=O)CC)CCN(C(c2cc(C3CC3)sn2)=O)CC1 C1(C(=O)NCCNC(c2ccnc(N3CCCC3)n2)=O)CCCC2C1C2(F)F C(N=c1[nH]c(N2CC3CC=CCC3C2)nc2ccsc12)C1(C)CC1 C1(C)(C(=O)NCC2N(C(c3cc(OC)ns3)=O)CCC2)C2CC3CC(C2)CC1C3 C1(C(=O)NCCOCC#C)CCN(C(=O)C=Cc2ccoc2)CC1O CN1CCOC2(CN(C(=O)C(C3(O)CCCCC3)NC(C3CC3C(N)=O)=O)C2)C1 Cc1cc(C(=O)NCC(N2CC3(C2)CN(C(C)C)C3)=O)ccc1[N+](=O)[O-] C=CC(CCC)CC(=O)N1CCC1C(=O)NCC1CCC(O)CC1 c1(OC)ccc(C(C)NC(=O)NC2CC(=O)N(c3c(F)cccc3Cl)C2)cc1F c1(C(CC)C)cccc(NC(c2cc(Cl)c(Cl)s2)c2nnnn2CCCF)c1 C1(NC(=O)C=CCO)CC(CO)N(C(c2cc(Cl)ns2)=O)C1 N#Cc1cccc(C2=CCN(C(=NCCN3CCSCC3)NC3CC3)CC2)c1 c1ccc2nc(NCC3SCCS3)c(NC3Cc4cscc4C3)nc2c1 C1(C(N2CCC(O)(CCNC(=O)C=Cc3ccoc3)C2)=O)CC(C2CC2)=NO1 c1(OC)cc(OC)cc(C(=O)NC2CC2NC(=O)Cc2cc(Cl)ccc2Cl)c1 c1(C(=O)OC)cccc(CNCC2CC2C(=O)NCc2ccnc(C)c2)c1O C(=O)(C(C)CCc1ccccc1)NCCOCCNC(COCC(=O)OC)=O C1(C)(CC)CCC(NC(=O)C(C)(C)CCNC(=O)C(c2ccccc2)C)CC1 N1(C(c2c(C#N)cn[nH]2)=O)CCC2(CCCN2C(=O)CC2CCC3CC3C2)C1 N1(C(C=C(C)Cl)=O)CCCC(C)C1CNC(c1csc(-c2ncc[nH]2)n1)=O N1(C(CS(=O)(=O)NC(C)(C)C)=O)CCCC2C1CCN2C(=O)CS(N)(=O)=O C1(C(=O)N(C2CC2)CC2CC2)(CNC(c2cc[nH]c2C2CC2)=O)CCCC1 c1(SC)cccnc1C(N1CC2C(CNC(=O)C(C)CSC)C2C1)=O c1(OC)cc(C(=O)NCC2(C)CCCN(C(c3sc(C)nc3C)=O)C2)ccc1C C(C(C(F)(F)F)NC(c1ccc(CN2CCCC(CN)C2)cc1)=O)NC(=O)NC N1(C(c2nc(C)oc2)=O)CCC2C(NC(c3cc(C(N)=O)cs3)=O)C12 CCC(C)CC(=O)NCC1(F)CCC(NC(c2ncccc2C(F)(F)F)=O)C1 C(N=c1cc(F)nc[nH]1)C1N(C(C2(F)CCCCCC2)=O)CCCC1 S(=O)(=O)(c1cccc(=NCC(O)CN(C)C)[nH]1)NCCOc1cccc(OC)c1 C1(NC(C(c2ccoc2)NC(c2cc(CC)no2)=O)=O)CC(C)(OC)C1(C)C c1(CNC(CS(CC)=O)=O)nc(CNC(=O)C(F)CC2CN(CC)C2)cc(O)n1 N1(C(c2c(COC)nn[nH]2)=O)CC(NC(=O)C=CSC)CC12CCC2 CCCCCC(O)CC(=O)N(CC(CC)NC(c1cccnc1)=O)C CC1CN(C(=O)CC2SC(=N)NC2=O)CCC1CNC(C1CC2C=CC1C2)=O C1(C(N(C2CC(NC(c3c(C)ncn3C)=O)C2)C)=O)Cc2ccccc2C1 c1(CC)cc(C(=O)NCC2CC3(CC3)CN2C(=O)C(CO)NC(N)=O)ccc1F c1(OCC)ccc(C(=O)NC(C)C(=O)NC(C)COC)cc1.c12csc(n1)O2 N1(C(CC)=O)CCN(C(=O)NCCc2cnn(C(C)C)c2F)C(C(C)C)C1 c1(CC(=O)NCC2COC(CNC(C3(CF)CCC3)=O)C2)n[nH]c2ccccc12 C(=O)(C1CCCc2cncn21)NC1(CF)CN(C(C(CCC)CC(C)C)=O)C1 C(=O)(C(CCC(=O)OC)NC(C)=O)N(CCNC(=O)CC1C=CCC1)CC c1(CC)cc(C(=O)NCC2CCC(NC(C3CC34CCCC4)=O)C2)sc1C C1(C(=O)Nc2c(C)cccc2)CCCC12CCN(C(=O)CCN(C)C)C2 CCCCC(O)CC(=O)NCC(CC(C)C)NC(=O)CCn1ccc(C)n1 c1(C(N2CC(N3CCN(C(C4(C)CC4(F)Cl)=O)CC3)C2)=O)cnc(Cl)cc1Cl CCC(C(=O)N1CCC(N(C(=O)CCOCc2ccccc2)CCO)C1)SC CC1(CNC(c2c[nH]nc2CNC(c2ccoc2)=O)=O)CCCC1O C1(C(N(CC(N)=O)C)=O)CC1C1CN(C(C2(F)CCOC2)=O)C1 c1(C(N2CCC(N3CCN(C(CC(CC)SC)=O)CC3)C2)=O)cc(C)cc(F)c1 c1(OC)ccc(C(C)C(N2CCCCC2CNC(c2ccn(C)c2)=O)=O)cc1F N1(C(C2(c3ccc(-c4c(SCC)ccc(F)c4)cc3)CC2)=O)CC2CCCCC2C1 C(=O)(C1=CS(=O)(=O)CCC1)NC1C(NC(C2CC(=O)NC2)=O)CC(F)(F)C1 C1(CNC(=O)Cc2ccccc2)CN(C(=O)CCN2CCCCCC2)CC12CC2 c1(C(=O)NC(C)CCCNC(=O)CC2CC=CC2)cc(F)c(Cl)cc1Cl N1(C(C2C(C=C)C2)=O)CCC2(CCN(C(c3ccc(OC)nn3)=O)C2)C1 c1(C(N2CC(NC(c3cncc(NC)c3)=O)C(C)C2)=O)ccc2c(c1)nnn2C N1(C(=O)OC(C)(C)C)CC(C(=O)O)(CCC(C)(C)N2CCCC2)C1 C(C(C)(C)C(=O)NCC#CCNC(c1cscc1-c1ccccc1)=O)N(C)C N1(C(C2C(CC)C2)=O)CCCCC1CN(C(=O)COC(C)=O)C C1(NC(=O)Cn2cc(SCC(F)F)nn2)CCCN(C(C2CCC(=O)N2)=O)CC1 N1(C(c2snnc2C)C(=O)NC(C(=O)OC)C)CC(=O)N(C)C(C)C1 c1(CC(=O)NC2CCC(Cn3cc(C(C=C)(C)O)nn3)C2)ccc2occc2c1 N1(C(CC2(C=C)CCC2)=O)CC(OC)C(NC(C2(F)CC2)=O)C1 CN1CCN(C(C2CCCC2c2nc[nH]n2)=O)CC1CNC(c1ccoc1Cl)=O C#CCCCC(=O)NCC1CCCC1NC(=O)C(C1CCOC1)OCC c1(CN(C)C(=O)NCc2ccc(Cl)cc2)cc(Cl)ccn1 C1(NC(c2ccc(CCC)s2)=O)CC2CCC(C1F)N2C(=O)C1=C(C)OCCC1 C1(NC(=O)Cn2ccnn2)CCN(C(C2(O)CCCC2)=O)CC12CCC2 CC1(CNC(=O)CC(F)F)CCN(C(c2ccc(CC3CC3)cc2)=O)C1 C1(CC(N2CC(CNC(C3(SC)CC3(F)F)=O)OCC2)=O)CCn2cncc2C1 C1(CNc2cc(NCC3COCCO3)ncn2)CC2CCCC2C1 c1(C(N2CC(CN(C(=O)C(F)(F)c3cnccn3)C)C2)=O)nocc1Cl S(=O)(=O)(c1ccc(NC2CCC(C(N)=O)CC2)c(F)c1)NC1C(C2C(C)C2)C1 C(=O)(CCCS(N)(=O)=O)NC1CCCC(CN(C(=O)CCCCC#N)C)C1 c1(C(C(=O)NCc2ccc(C3(C)CC3(F)F)cc2)F)c(F)cccc1F C1(NC(=O)CN(C(=O)CCCn2cncn2)C(C2CC2)C2CC2)COCC1CO c1(-c2onc(-c3c(CC)ccc(O)c3)n2)c(F)ccc2ccoc12 C(=O)(CCCCC(C)(C)C)N(C1CCCC(N(C(c2ncn(CC)c2)=O)C)C1)C N1(C(C2C3CC4C(C3=O)C24)=O)CC2CCOCC2(NC(C2(F)CCCCC2)=O)C1 c1(CCNC(C(N2CCN(C)C(C(F)(F)F)C2)=O)=O)csc2ccc(Br)cc12 N1(C(CC(C(C)C)O)=O)CC(C)(CNC(c2cncc(CO)c2)=O)CC1(C)C Cc1onc(-c2ccsc2)c1C(=O)NCCN(C(=O)C(c1ccc(Cl)s1)C)CC C1(NC(c2c(COC)cccc2)=O)CCN(C(=O)CN2CCSCC2)CC1(C)C C(=O)(CC(C)C(C)(C)NC(=O)C(O)C1CCCC1)NCc1n(CCC)ncn1 N1(C(CC2(C=C)CN(C(=O)CC(CC)C(F)F)C2)=O)CCN2CCCCC1C2 Nc1cnc(Cl)c(C(N2CC(CNC(c3c(Cl)csc3Cl)=O)C2)=O)c1 c1(OCC)cccc(C(=O)NCC23CC(C2)C(NC(=O)CCF)CO3)c1N C(CC(C)C)(C(=O)NC(C)(CNC(c1cnc(C)[nH]1)=O)C1CC1)OC C1(CNC(C23CC(n4cc(C5CCCC5)nn4)C2C3)=O)CCS(=O)CC1 c1(CC(=O)NCCC2OCCN(C(C(C=C)O)=O)C2)nc([N+](=O)[O-])n[nH]1 Cc1cnccc1C=CC(N1CCC(CO)(NC(c2ccc(F)s2)=O)CC1)=O C1(CCNC(=O)Cn2cccn2)CN(c2ccncn2)CCS1(=O)=O CCC(C)C(C(=O)N1CCCC(C(N2CCC2C(=O)OC)=O)C1C)N(C)C c1(OC(C(C)C)C(=O)NCc2cnn(C3CNC3)c2)ccccc1[N+](=O)[O-] CC(C)(C)S(=O)(=O)c1ccc(=NCCCOCCOCCOCCO)[nH]c1 C1(C(N2C(C(=O)NCC#CCC)C3CC3C2)=O)CCOC(C)(C)C1 c1(C(=O)NC2CC(NC(CCC)=O)C23CCC3)cc(Br)c(C)cc1O CC1(C)C(NC(c2c[nH]c(C(N)=O)c2)=O)CC1O CN=c1nc(N2CCc3cccc(C)c3C2)[nH]c(=NC2CSC(C)C2)[nH]1 c1(CCC)nc(C(=O)N(CC(C)N(C)C(c2coc(Br)n2)=O)C)cs1 C(CCO)(C(F)F)N(C(c1c(CNC(C(C)O)=O)noc1)=O)C C(c1ccccc1OCC#N)=CC(=O)NCc1cnn(CC)c1C Cc1c(C(=O)NCC2C3CN(C(c4cn(C)nc4O)=O)CC23)cncc1F c1(C(=O)NCC2(F)CCC(NC(C=C(CCC)C)=O)C2)cn2c(C)csc2n1 CC1CCC(CCNC(=O)CCN(CCCO)C(C2(C)CC(C)C2)=O)CC1 Cc1nc(C(N2CC(C)CC2(C)C)=O)c(F)c(Cl)n1 N1(C(c2c(Cl)ccc(OC)n2)=O)CCOC2CN(C(c3ccsn3)=O)CC12 c1(C(N(CCN(C(CCN(C)CC)=O)C(C)C)C)=O)ccc([N+](=O)[O-])nc1 Cc1cc(C(=O)NCc2nnn(C(C)(C)C)n2)c(C)nn1 CC1CCN(C(c2cncc(NCc3cncc(Cl)c3)c2)=O)CC1NS(C)(=O)=O c1(C(=O)OC)nccc(C)n1.N1(CC)CCC1C(=O)NC C1(C)(COC)CC(NC(c2oc(CO)nc2C)=O)CN1C(C1CN(C(C)=O)C1)=O C1(C(=O)NCC(CCCC)NC(c2cc(O)nc(O)c2)=O)CCC2CC2CC1 c1(C(=O)NCCN(CCC)C(C2CC2C(C)C)=O)csc(C)c1 N1(CC(COCC(C)C)O)CCCC2C(NC(=O)CCc3cscn3)C(C)(C)C12 C#CCC(C(=O)N1CC(C)(OC)C1)NC(c1cc(Cl)cs1)=O C=CC(CC)CC(=O)N1CC2(CC(NC(=O)C(CCC)NC(C)=O)C2)C1 Cc1nn(C)cc1CCC(=O)N(CCNC(c1cc(C2CCC2)on1)=O)C1CC1 C1(C)(NC(C(c2ccc(F)cc2)SC)=O)CCN(C(c2cc(F)c[nH]2)=O)C1 C(CCCC(C)NC(C1CCCO1)=O)NC(c1c(CC)cno1)=O C(=O)(CCc1ccno1)NC(C)CN1CCCC1 C1(O)(C(C)NC(C2(C)CC2C(F)(F)F)=O)CCN(C(C2SCCS2)=O)CC1 n1(C(C)C)nccc1C(=O)NCC1(CNC(=O)C(C)(C)n2cccn2)CCC1 c1(C(=O)OC)cc2cc(C(=O)NC3CCCC3n3cc(C4(C)CC4)nn3)sc2s1 CCCC(CC)CC(=O)NCCC1CC(NC(=O)Cc2scnc2C)C1 CN1CCOC2(CN(C(C34COCC3CN(C(=O)CC(C)(C)O)C4)=O)C2)C1 C1(NC(CC2(OCC)CC2)=O)CCC12CCN(C(=O)CC(C)(O)C(F)(F)F)CC2 c1(COCC)nc(Cl)cc(=NCC(C)NC(C2COc3ccc(F)cc3C2)=O)[nH]1 C1(OC(C2C(OC)CC2)=O)CCCN(c2cc(C)ccc2Cl)C1=O C(=O)(C1COc2ccc(Cl)cc21)NCCC1CCCN(C(C(C)(F)F)=O)CC1 N1(c2c(CC)c(Cl)ncn2)CC2CCC1C1CN(C(C3CCC(F)C3)=O)CC21 c1(OCC)ccccc1-n1cc(CN(C)C(c2sc(C(F)F)nc2Br)=O)nn1 C1(F)(C(=O)NCCC2C(C)(C)OCC2)CCCN(C(C2CCCCC2(C)C)=O)C1 CC(C)CC(C)(O)CNC(=O)C(C)NC(=O)CCSCC(N)=O c1(OC)cc(C(=O)Nc2cc(-c3ccnn3C)ccn2)cc(Br)c1OC c1(OC)c(C(=O)NC2CN(C(C3CCCCC3)=O)CC2C(F)(F)F)ccnc1Cl N1(CC(=O)N(C)CC2C3CN(C(C4CC45CC5)=O)CC23)Cc2ccccc2C1 c1(C(=O)NC(C(C)C)CCN(C)C(C2(N(C)C)CC2)=O)cn(C)c(=O)nc1O C12(C(=O)NCCC(=C)CNC(C3(C)CCC3)=O)CC3CC(CC1C3)C2 c1(OCC)ccc(C(N2CCC(CNC(c3ccnc(C(N)=O)c3)=O)C2)=O)cc1 c1(N2CCN(C(C(c3cccc(F)c3)C)=O)CC(O)C2)ccc(Cl)cc1[N+](=O)[O-] C1(CC)CCN(C(=O)C(F)C(C)(F)F)C(C(=O)NC2CC23CCOCC3)C1 C12(NC(c3ccnc(CO)c3)=O)CC3CCC(C1C2)N3C(=O)Cc1ccsc1 C(CNC(C1(C2CCCCO2)CCC1)=O)(CC(F)(F)F)NC(CCCCOC)=O C(C1(C)CCC(C)C1(C)C)=CC(=O)NCC1COCCN(C(C(C(C)O)C)=O)C1 N1(N(C(=O)Cc2nnn(C(C)(C)C)n2)Cc2n(CC)nnc2)CCc2ccsc2C1C C1(COC)(NC(c2ccc(F)cn2)=O)CCN(C(C2CC(n3ccnc3)C2)=O)C1 C1(NC(C2(O)CN(C(=O)CSCC(N)=O)C2)C)CCN(C(=O)C(=O)N(C)C)CC1 C1(NC(C2C3(CC(C)(C)C3)C2)=O)CCCCC12CCN(C(C1(F)CCOC1)=O)C2 c1(C(N2C(C)C(NC(=O)CC(C)C(F)F)CC2)=O)nn(C)c2c1CCC2.C(C)(C)C c1(C(C(=O)NC2CCOC2)N(CCCOC)CCOC)coc(Br)n1 Cc1c(C(N2CCC(C)C(N(C)C(C3CCC3)=O)C2)=O)[nH]c2ccccc12 c1(C(N(C)CC2(NC(c3csc(-c4cnccn4)n3)=O)CC2)=O)cscc1F CC(CF)CC(=O)NC(C)CC(C)NC(=O)C(=O)NC1CCCCC1 CC1CCN(C(=O)CC2CCCCC2)CC1NC(=O)CCc1ncc(F)cn1 CCC(C)CCCC(=O)NCC(C1CCC1)NC(c1sccc1-n1cccc1)=O C1(CNC(CN(C2CCC2)C)=O)C2CN(C(=O)CCN3CCCS3(=O)=O)CC12 CCC(O)C(C)C(=O)NC1CCN(C(C2CN(c3nncs3)C2)=O)CC1F C(=O)(C(F)C(C)(C)O)NCC(CNC(c1c(C)nn(-c2cnn(C)c2)n1)=O)CO c1(NC2CN(C(C3(C=C)CCC3)=O)C2)nc2c(cc1C#N)CCC2 N1(C(C2CCC3(CCC3)CO2)=O)CCN(C(=O)Cn2cc(Cl)cn2)C2(CCC2)C1 C1(OCC)CCCCC1C(=O)NCCCN(C(=O)C(C)NC1(CO)CCCC1)C Cc1ncnc(C(=O)NC2CN(C(=O)C(C)(F)F)CC2C)c1C C1(CNC(C2(CC)CC2(F)F)=O)CCN(C(c2cnccc2N(C)C)=O)CC1 CC(C)(C#N)CCCC(=O)N1CCC(C(=O)NC2CC3C(C2)C3(F)F)C1 C12(C(N3CC(O)(CNC(=O)C(O)C4CCCC4)C3)=O)CC(C1)S(=O)(=O)C2 C=CC1COCCN1C(C1CC1C1CN(C(=O)CCCCOCC)C1)=O N1(C(C2CCC(N(C)C)C2)=O)CCC2CCCC12C(=O)NCCn1cccnc1=O C(CCCC(C)NC(c1cccc(=O)o1)=O)NC(c1c(C)cns1)=O N#CCCCCC(=O)Nc1cccc(CNC(=O)C=CCCc2ccccc2)c1 N1(C(C(C)NC(C)=O)=O)CC(C(=O)Nc2ccc(C(F)(F)F)nc2Br)C2(CC2)C1 C=CCC(CC)C(=O)N1CCN(CCNC(c2ccc(CC3CC3)cc2)=O)CC1 C(=O)(C(C(=O)OC(C)(C)C)C(C)(C)C)NC1CC(C)(NC(C=C(CCC)C)=O)C1 c1(-c2n(-c3cnc(C)s3)nc(C3CCCO3)n2)ccc2nc(Cl)nn2c1 c1(NCc2cnc(COC)[nH]2)cc(N2CC3CC3C2)nc(COC)n1 N#CC1CC2(CC(C(=O)NCCCc3nc4ccccc4[nH]3)C2)C1 c1(CC(=O)NCCOCCNC(C(C)(C)C2CCCCO2)=O)c(O)ncnc1O N1(C(CN(CCC)C)=O)CCC(C)(C)C(NC(C2CN(C)C(=O)CCO2)=O)C1 C=CC(C)(O)CC(=O)NCCN(C(=O)C(CCC)NC(C)=O)CCC C12(CC)CCC(C(N3CC4(C3)CN(C(c3ncn5c3CCC5)=O)C4)=O)(CO1)C2 C(=O)(C(C)S(C)(=O)=O)NCCn1cc(C(N(C(CC)C)C)=O)nc1 C#Cc1cccc(C(C(=O)NC(C)(C)CC)N(C)C(c2ccco2)C)c1 C1(F)(CNC(C(C)NC=O)=O)CCN(C(c2ccc(Cl)cc2)=O)C1 N1(C(CC2(C)N(C(C(CCCC)O)=O)CC2)=O)CCc2cccc(F)c21 CCN=c1[nH]c(C(=O)NC(C2CCN(C(c3sc(N(C)C)nc3Cl)=O)C2)C)cs1 C12(CNC(c3n(CCOC)nnn3)c3occc3C3CC3)CCCCC1CCC2 c1(C(C)C(N2CC3CC3(CNC(c3cc[nH]c3)=O)C2)=O)cn(C)c2ccccc12 Cc1nn(C)c(C)c1CC(=O)NC(C)CCCNC(=O)CN1OC(C)(C)CC1=O C1(NC(c2ccc(Br)c(F)c2)=O)COC2(CCN(C(=O)CO)CC2)C1 c1(C(=O)OC)cc2c(N(C3C(F)(F)C34CC4C(=O)OC)C)ncnc2n1C C1(C(C)NC(CN(C)CC)=O)CC(NC(c2ccon2)=O)C1 c1(C(C(=O)NCC)N(C(c2ccncc2Br)C(=O)OC)C)nccc(Cl)c1F CC(C(=O)N1CCC(OCCNC(=O)C(C)(O)c2ccccn2)C1)S(N)(=O)=O c1(C(N2CCC(CNC(=O)CCc3cscn3)C2)=O)noc2c1CCCC2 C(=O)(C1=C(F)CN(C(=O)C(C)C2CCC2)CC1)NC(c1c(C)nn(C)c1)C c1(CNC(C(=O)NCCCOC)=O)ccc(Br)cc1OC(F)F c1(C(C)C)c(N2CC(CNC(C3CCC4CC34)=O)C(C)C2)ncnc1Cl n1(C(C)C)nccc1C(=O)N(CCCN(C)C)CCNC(c1ccc(CO)o1)=O c1(C(N2CCC(NC(C3(O)CC(F)(F)C3)=O)CC2)=O)ccn2c(O)nnc2c1 CC1CCC(F)(F)CN1C(=O)CC1(C)CCN(C(=O)Cc2cn[nH]c2)C1 c1(C(C)(C)C)ccc(CCC(=O)NCC(O)CNC(=O)CC2CCCCO2)cc1 C(C(C)(C)CC(=O)N1CCCC1(CC(C)C)C(=O)O)OC C1(C(C)NC(C(C2CCCC2)NC(C)=O)=O)CN(C(C2(O)CCCC2)=O)CCO1 c1(CC)ccccc1C(N1CCC(O)(CNC(=O)CCc2ccsc2)C1)=O c1(C(C)=O)cccc(N(Cc2cccc(Cl)n2)CC2CCOCC2)c1 N1(C(C(C)OCC2CC2)=O)CCc2ccccc2C1CCNC(C1CC1(C)C)=O N1(C(CC(C)(C)c2cccs2)=O)CCN(C(=O)COC2CCC2)C2CCCC12 c1(NC(C(=O)NC(c2ccc(F)cc2)(C(=O)OC)C)C)cccc(C#N)c1 c1(N2CCOCC(C)(F)C2)nc(NC2CN(CC(F)F)C2)c2ncsc2n1 N1(C(=O)C2=CCCCC2)CCC(NC(C23CCCN(CC2)C3)=O)C(F)(F)CC1 N1(C(C2C=C(C)CS2)=O)CC(CC(=O)NCC(=O)NCC2CC2)CC1(C)C c1(C(=O)NCCC2CC(NC(c3cc(C(F)F)cs3)=O)C2)occ2c1CCC2 c1(C(=O)NCCC(CNC(=O)Cc2csc(S)n2)O)cnn2c1CCC2 Cc1nccc(C(=O)NCC(O)CN(C(=O)COCC2CC2c2ccco2)C)n1 CC1ON=C(C(=O)NCC2(C)CN(C(=O)CCP(C)(C)=O)CCO2)C1C C1(NC(c2c(CC)n[nH]c2)=O)CCC(F)(CNC(c2cncc(C(F)F)c2)=O)C1 C1(C)(OCC(=O)NC2C(NC(C3(CC=C)CC=CC3)=O)CC2)CCOCC1 N1(C(C2C(OC(C)=O)C2)=O)CCC1(C)CC(=O)NCc1nc(N(C)C)n[nH]1 CC1(C)CC(CNC(c2cccs2)=O)CN1C(C1CCCC1(F)F)=O c1(-c2cn(C3C(C)CCN(C(=O)OC)C3)nn2)cc(C(=O)O)c(F)c(F)c1 Cc1[nH]nc(C(=O)NCC2CC(F)(CNC(C3(C)CC3C(F)(F)F)=O)C2)c1Cl C(CC(F)F)(C(=O)N1CC(C2(C)CC2)C1)N(C(C(C(=O)OCC)F)=O)C CCC(CC(=O)NC1CC(CNC(=O)CCCC2CC2)C1)C(=O)OC(C)(C)C C(=O)(CCCCCOC)NCC(c1ccc(F)cc1)NC(CCC)=O c1(C(N2CCC(C(C)CNC(=O)Cc3cn[nH]c3)CC2)=O)cccc2ccoc12 N1(c2cc(N(C)C)ncn2)CCC(NC(c2cn(CCO)nn2)=O)C(F)C1 c1(C(=O)NCC2CCN(C(C3(NC(N)=O)CC3)=O)CC2O)cccn2cnnc12 Cc1cccc2c(C(N3CC(C4CN(C(c5ccnnc5O)=O)C4)C3)=O)c[nH]c12 C1(CNC(c2n(C)c(S)nn2)=O)CC2(CCC2)CN1C(=O)CC1(C)CC1(Cl)Cl C1(C(N(C(CC)C2CC2)C)=O)CCOCC1NC(=O)CCOCCOC C1(COC)(CNC(C2(C)CC=CCO2)=O)CCCN1C(=O)C(C)=C(C)C c1(CC(N2CC(NC(C=C(C)Cl)=O)C3(C2)CC3)=O)ccc2oc(O)nc2c1 c1(C(=O)NCc2c(C(=O)NCC(C(N)=O)O)nco2)cc2occc2[nH]1 N1(C(C(N2CCNC2=O)C)=O)CCC2(CCCC2CNC(=O)CCC(F)(F)F)CC1 C1(C(=O)NCC2CN(C(C(C)Oc3cccc(Cl)c3)=O)C2)CCC(C)(F)CC1 c1(C(=O)NC2CN(C(C3(F)CC(C(=O)OCC)C3)=O)C3C2C3)ccc(Cl)cc1Cl CC(CCC(=O)NC1CC(CNC(C2(n3cccn3)CC2)=O)C1)c1ccccc1 c1(C(=O)NCC(C)NC(C(CC#C)O)=O)ccc([N+](=O)[O-])c(OC)c1 C(CCSC)(C(=O)N1CC(CNC(=O)CCSCC(N)=O)(OC)C1)OC N1(C(C(C(COC)C)C)=O)CC2CCCC(NC(=O)Cn3nc(C)oc3=O)C2C1 CCCCC(O)C(C)C(=O)N1C2CCCC1CN(C(=O)C(O)Cc1cnc[nH]1)C2 C1(C(=O)NC(CCCNC(c2c(C)nc(C)s2)=O)(C)C)CCOC2(CCCC2)C1 c1(NC(CSCC)=O)csc(C2CCCC2)n1.C12CCCN1CC(=O)NC2 CN(C)S(=O)(=O)N1CCC(C(=O)NC2(C)CCCN(C(=O)C=C3CC3)C2)C1 C(C(C)(C)C(=O)NCC1CCN(C(=O)Cn2cc(-c3ccccc3)nn2)C1)SC C=CCC(C(=O)NC1CC12CC(NC(c1ccccc1C#N)=O)C2)C(C)C c1(OC)cccc(C(=O)NC(CNC(=O)C(c2cccnc2)C)CO)c1 CC1CCC(NC(=O)CCCC(N)=O)CN1C(=O)C=CCCc1ccccc1 C(C(C(=O)NCC1CC(O)C1(C)C)C(C)(C)C)NC(C(C)C(F)F)=O C12(NC(c3ncccc3Cl)=O)CCN(C(c3csnn3)=O)CCC1C2 N1(C(c2ccc(C)nc2C)=O)CC(NC(=O)C(C)c2ccco2)C(C2CC2)C1 C1(CC(=O)NCC2CCN2C(=O)CCc2ncc[nH]2)CC2(CC2)C1 C1(CC)(NC(c2nc(C(C)(C)C)no2)=O)CCN(C(c2cnc(C)[nH]2)=O)CC1 CC(C(=O)N(C)Cc1cn(C2COC(C)(C)C2O)nn1)C(F)(F)F N1(C(c2c(C)ccc(C(N)=O)c2)=O)CCC2(CC1)CN(C(C1CCC1F)=O)C2 CCCC(C(O)C(=O)N1CCC(c2nc[nH]n2)C1)NC(C1(C)CC2CCC1O2)=O CS(C)(=O)=NCC(=O)NC1(CO)CCCN(C(=O)CC2CC3(CCC3)C2)C1 c1(C(N2C(C3CCN(C(C(=C)F)=O)CC3)CCCC2)=O)cc(F)c(Cl)c(F)c1 c1(CNC(COc2c(C)cc(C)cc2C)=O)cc(=O)n2nccc2[nH]1 c1(OC)cc2c(cc1C(OC1CCc3cc(Cl)ccc31)C(=O)NC(C)C)OC(C)C2 C(=O)(CCCC(C)C)NC(CC#C)C(=O)NCc1nccc(OC)n1 C1(C(N2CC3(CC(NC(C=C(CCC)C)=O)C3)C2)=O)OCC2CCCCC12 N1(C(C2(CC=C)CCC2)=O)CC2CN(C(c3cnc(C)s3)=O)CCC2(CO)C1 c1(C(N2CCN(c3ccc(NC(C4C(C)C4)=O)cc3)CC2)=O)cc(Br)cnc1O C1(NC(=O)CC2CC2(Cl)Cl)CCN(C(c2cc(Br)co2)=O)CCC1CO N1(C(CC2C(C)=NN(C)C2=O)=O)CCN(C(=O)C2=COCC2)CC(C)(C)C1 CC(N=c1nc(N2CCn3nc(C4CC4)cc3C2)c2c([nH]1)CCS2)C1CCC1 N1(C(Cn2c(=N)[nH]nc2)=O)CCCC(O)(CNC(=O)COc2cccnc2)CC1 c1(OCC)ccc2c(c1)CCCN2C(c1cnn(CCO)c1C)=O C1(NC(c2ccc(SC)s2)=O)CCCC(NC(=O)CCS(N)(=O)=O)CC1 C(C(CO)(CO)CO)NC1CC(C)OCC1 C1(NC(CCCCN(C)C(C2COCCO2)=O)=O)CC2CC1OC(=O)N2 c1(OC)nc(C)ccc1CNc1cc(-c2nn[nH]n2)ccn1 C(C(C)(O)CC(=O)N1CC2CC1(C(=O)Nc1ccccc1C(C)C)C2)OC c1(CC(=O)NC(C2CCCCC2)C(=O)N(C(C=C)C)C)cc(C)on1 c1(C(=O)NCC2CN(C(C3(C)C(C)OCC3)=O)C2)c(Cl)cc([N+](=O)[O-])cc1Cl Cc1nn(C)c2sc(C(=O)N(CC(C)(C)CNC(=O)CC(=O)NC3CC3)C)cc12 CC1(C(=O)NC2(C(=O)NCCc3nccc(O)n3)CC2)CCC(=O)N1 C1(C(=O)NC2(c3ccccc3)CN(C(c3c(CC)nc[nH]3)=O)C2)CCCC(C)C1 CCC(CC(=O)N1CCC(O)(C(C)NC(c2csc(O)n2)=O)C1)C(C)(C)C c1(C(N2CC(C)C(CNC(C3COC4(CCC4)C3)=O)C2)=O)c(N)cccc1F C(=O)(C1=CC2(CCOC2)C1)N1C(CN(C(c2cccc(Cl)c2Cl)=O)CC)CCC1 c1(C(N2CC(CC(C)NC(COCC=C)=O)C2)=O)ccc(C2CC2)cc1Cl C=C(C)CC(C)C(=O)NCc1ccc(CNC(C2(CCO)CC2)=O)cc1F Cc1nc2c(C(N3CCOCC3CNC(C3CCS(=O)(=O)C3)=O)=O)ccnc2[nH]1 CC(C)C(C)(CNC(=O)CSC1CC(C)N(C)C1)NC(c1ccsc1)=O N1(CCC#C)CCN(C(=O)CC2CN(C(C3CC34CCC4)=O)CC2C)CC1 c1(C(c2n(CCCC)nnn2)NCC2COCCO2)cncc(Br)c1C CC(C)CC(C(=O)NCC1(C)CN(C(c2cc(Cl)no2)=O)C(C)(C)C1)C(N)=O CC1(C)OCC2CC12C(=O)NCCCNC(=O)Cc1cn[nH]c1 c1(C(C)NC(=O)C=CCNC(C2(C(N)=O)CCC2)=O)cncnc1 c1(C(=O)NCC=CCNC(CC2C(C)CCO2)=O)cc([N+](=O)[O-])cn1C CCC(CNC(=O)C(c1cccnc1)NC(c1cc(Cl)cn1C)=O)C(C)(F)F c1(-c2cn(-c3c(C(N4CCCC4CCCO)=O)scc3)nn2)cnc(O)nc1 n1(C(C(=O)N(C(CNC(CNC(=O)OCC=C)=O)C)C)C)nc(C)cc1C c1(C(C(C)OC(C(COC)(C)C)=O)=O)cc(C)n(C(C)C(=O)OC)c1C CC1CCN(CCC(=O)NCC2(F)CC(NC(C3CC(CCO)C3)=O)C2)CC1 C(CCCCCC(=O)NC1(CO)CC2CCC1C2)NC(C(C)SC)=O C1(NC(c2c(OCC)nccc2)=O)CCN(C(=O)C(C)C(C)C)CC1(C)C C1(N(C(C(CC2CCCC2)NC(CCCOCCC)=O)=O)C)CCCC(C)C1C N1(C(C2CCC2)=O)CC2CN(C(c3cccc4nc[nH]c34)=O)CCC2(CO)C1 N1(C(Cc2c(CC)con2)=O)C(CNC(C2CCC2C(=O)OC)=O)CC2CC12 c1(C(=O)NC2(CNC(C3C(C)(C(C)C)C3)=O)CCC2)nccnc1N C1(C(=O)NC(C)CNC(=O)CSCc2cccnc2)CCNC(=O)C1 c1(OC)ccc(Br)cc1C(N1CCC(C)(C(=O)NCC2(C)CC2)C1)=O C(C1(O)CCc2ccccc21)NC(=NCC=C)NCc1conc1CC Cc1nc2ccc(N3CCCC3c3ccncn3)nn2c1I c1(C(N2CCCC(C(C)NC(c3cncs3)=O)C2)=O)ccc(N)cc1Br C(C)(CNC(=O)CCSc1ccccc1F)(C(C)C)NC(C1C(C(=O)OC)C1)=O c1(C(=O)NC2CN(C3CN(C(CC4(C=C)CC4)=O)C3)C(=O)C2)cc(F)ccc1C c1(NC(CCC)=O)ccc(NC(=O)Cc2ccc(Cl)c(OCC)c2)c(C)c1 C1(NC(C(C2(C)CC2)NC(C2CCCCCC2)=O)=O)CCOC12CCCC2 Cc1ncoc1C(=O)NC1(CCNC(=O)C(=O)Nc2ncc[nH]2)CC1 C1(C)(OC)CCCN(c2nnc(CC(C)C)n2CC2CCOC2)CC1 C1(C(=O)C)CCN(C(=O)C(N2CCCC2C(C)(C)O)=O)CC1.CO c1(C(=O)NC2CCCN(C(=O)Cn3cnc(Br)c3)CC2)ccc2ccoc2c1 c1(C(N(CCOCCNC(c2cc(C)[nH]n2)=O)C)=O)c(Cl)ccc2c[nH]nc12 c1(-c2nnc(N(CCC#C)C)n2CC(=O)NCCO)nc2c(s1)COCC2 CC1CCC(C(=O)NCCCP(C)(C)=O)N(C(=O)CCc2ccnn2C)C1 N1(C(c2c(C)nsc2)=O)CCOCC(C(=O)NC2CCC3(CC3)C2)C1 C12(NC(CCCC)=O)COC(CNC(=O)C(C)SCCCC)(C1)C2 C1(C(=O)NCC2CCN(C(=O)CC3OCCO3)CC2)CCC2(C1)CC2(F)F N1(CC(=O)NCC(C)(O)CNC(=O)C(O)C2CC2)C(=O)c2ccccc2S1(=O)=O c1(C(=O)NC2C3CN(C(C4CC(C)(C)C4)=O)C2CC3)coc(S(N)(=O)=O)c1 COn1cnc(C)c1C(=O)NC1CC2(C1)CN(C(C1CC13CCOCC3)=O)C2 c1(C(c2n(CCCSC)nnn2)NC2CC(CO)C2)cnc(C(C)C)nc1 N1(C(C(CC2CN(C(C3(C)CC3)=O)C2)F)=O)CCC2(CSC2)C1 C1(NC(C(C)OCC=C)=O)CC2CC1CN(C(C1(CF)CCC1)=O)C2 O(NC(=O)C(CO)NC(=O)C(O)CSC(F)(F)F)CC(C)(C)O N1(C(C(c2c(C)cccc2Br)NC(=O)OC(C)(C)C)=O)CCCOCC1(C)C N1(C(CNC(CCC)=O)=O)CC2C(NC(C3(C)CCCO3)=O)C2C1 CS(=O)CCC(=O)NCC(C1CCCCC1)NC(c1cnc(C(C)(C)C)s1)=O c1(OC)ccc(CCNc2oc(COC(=O)C(c3ccc(Cl)s3)C)nc2C)cc1 C1(NC(c2ccc(C)s2)=O)Cc2ccccc2N(C(=O)CCC2CCC(C)O2)C1 N1(CC)CC(C(N2CCCC(N(C(=O)Cc3nocc3C)CC)C2)=O)CC1=O N1(C(COCC=C)=O)CC(C)(C(=O)NC2CC(CCC(N)=O)C2)C1 N1(C(C(COC)N(C)C)=O)C2CCC(C2)C1CC(=O)NCCCC1CCCC1 Cc1ccc(C)c(OCC(=O)NC2CC23CC(NC(=O)Cc2ccon2)C3)c1 C1(C(=O)NCC2(C(C)NC(C(C)c3ccon3)=O)CC2)CCCCC1 c1(OC)ncc(C(=O)N(CCCCN(C)C(C2CCOC2C2CC2)=O)C)cc1C CC(c1ccc(F)cc1)=CC(=O)NCC(C1CC1)NC(c1cc(O)cc(Cl)c1)=O C=CC(CCC)CC(=O)N1CCC(N(CCOC)C(C2CC=CCC2)=O)CC1 Cc1ccc(C(F)C(=O)NCC2(F)CC(CNC(c3ccc(C)nc3)=O)C2)cc1 Cn1cc(C(=O)NCC2(NC(C3C=CCS3)=O)CCC2)cn1 c1(CC)ccc(C(N2CCC(N=[N+]=[N-])C2)C(=O)NC)c(C)c1 N1(C(c2cnc(CCC)s2)=O)CCC12CN(C(c1cscc1C(F)F)=O)C2 c1(OC)ccc(C(=O)NCC2CC(C(=O)N(C(CF)CF)C)C2)s1 N1(C(c2ccn(CC)c2C)=O)CC2(C1)CN(C(c1cccc(O)c1F)=O)C2 c1(CC(N2CCC(N(C(c3ccn(C(C)(C)C)n3)=O)CCO)C2)=O)ccc(F)c(Br)c1 C(=O)(C(C)C(C)(C)C)NC1CN(C(c2nc(C)n(-c3ccccc3)n2)=O)CC1C Cc1c(F)ccc(-c2nc(NCc3ccc(N4CCOCC4)cc3)cs2)c1F c1(C(=O)OCC)cccc(S(=O)(=O)NC(c2ccccc2C)C(C)(C)C)c1 C1(C2CC2)(C(=O)NCC2(F)CC(NC(C(C)C(C)(C)C)=O)C2)CCOCC1 CC1(CCC(=O)NC2CCN(C3CC3)CC2)CCCN1C(C1CCOC1(C)C)=O N1(C(c2cncc(OC)c2C)=O)CC2CCC(CNC(c3cnsc3C)=O)C2C1 C(CCCC)(CCC)(c1nnnn1C1CC1c1ccco1)NCC1CC(SC)C1 N1(C(C2N(C(CCC(=O)NC)=O)C(C(C)C)CC2)=O)CCc2oc(C)nc2C1 C1(CCCC)CCC(NC(C2(CNC(c3c[nH]nc3C(F)F)=O)CC=CC2)=O)C1 C(=O)(C(C)C(F)(F)F)NCCC(CC)(C)NC(C1CC=CCO1)=O C=CC1(CC(=O)N(C)CC2CCCC(OC)C2)CN(C(c2cnc[nH]2)=O)C1 C(=O)(CCCCC(F)F)NC1CC(F)(CNC(C(C)Sc2ccc(C)cc2)=O)C1 C1(CC)CN(C(=O)CNC(=O)OC(C)(C)C)CCC1NC(c1cc(Cl)c[nH]1)=O N1(C(CCOCC#C)=O)CC2(CCN(C(=O)CC(C)C(C)C)C2)C1 CC1CC(c2cn(CCc3nccs3)nn2)CCN1C(C1CCO1)=O C1(NC(c2cnn(CCO)c2)=O)CC(F)CN(C(=O)COc2cccc(Cl)c2)C1 N1(C(CCC2CCC(C)O2)=O)CCOC2(CCC(Nc3ccncn3)CC2)C1 CC1CN(C(C2CCCC(O)C2)=O)CCN1C(=O)C1=CCSC1 c1(NC(N2CCOC(Cn3ccnn3)C2)=O)ccc2nc[nH]c2c1 N1(C(CCC(=C)C)=O)CCC(C(=O)OC)C12COC2 N1(C(C(c2cccc(OC)c2)O)=O)CCCC(N=c2nc(OC(C)=O)[nH]s2)C1 Cc1scc(C(N2CCCC2(C)CNC(=O)CC2CCC(C)CC2)=O)c1N CNS(=O)(=O)NCC(=O)NCCN(C(=O)C(C)(C)OC)C1CCO1 c1(OCCN2CCCC(NC(=O)C(F)(F)F)C2)cc2c(cc1F)CCC2NCC c1(NC(C2(O)CCN(C(C=CC(C)C)=O)C2)=O)ccc(F)c(Br)c1O C12(CNC(C34CC(C)C3C4)=O)CC1CN(OC1CC(C(=O)OC(C)(C)C)C1)C2 N1(C(c2nc(CNC(C(C(C)C)SC)=O)oc2)=O)CCN(C)CC1C C(=O)(C1=NN(CC)C(=O)CC1)N1CCC2C(NC(c3c(SCC)nccn3)=O)C21 N1(C(C(=O)NCC)=O)CCCC2CCN(C(=O)CC(=O)N(C)C)CC12 c1(C(=O)NCC2N(C(C3C(C(C)C)C3)=O)CC(O)C2)cc2n(n1)CCO2 c1(C(=O)NC2C(NC(CCC(C)(C)OC)=O)COC2)cn2cccc(F)c2n1 C1(NC(CC(C)c2cccnc2)=O)CCOCC1NC(=O)CCn1cccn1 N1(C(C(CCC)C)=O)CCOCC(C)(CNC(=O)CCSc2nccn2C)C1 Cc1ccc(Cl)c(OC(C)C(=O)NCC2CN(C(=O)CC3(CO)CC3)CCO2)c1 N1(C(C(CC)C#N)=O)CC(NC(=O)C(c2cccc(Cl)c2Cl)(F)F)CC1(C)C CC(C)(C(=O)NCC1(O)CC(CNC(=O)C=C(Cl)Cl)C1)C1CCCCO1 COn1cnc(C)c1C(N1CCC(CN(C)C(C2CC2C#N)=O)C1)=O CC1CCCN(C(=O)C(F)n2cccn2)C1CNC(=O)C=Cc1nccs1 C1(NC(C2CN(S(C)(=O)=O)C2)=O)CC2CC(NC(=O)Cc3ccsc3)C1C2 C(CC(=O)N1CC(NC(c2csc(O)n2)=O)C2(CC2)C1)(C1=CCCC1)OCC c1(CC(C)C)c(C(=O)NC23CC2CN(C(=O)CC=C(Cl)Cl)C3)cnn1C CC#CCC(C(=O)N1CC([N+](=O)[O-])C1)NC(c1cncn1C)=O C(CCC(=O)NCC1CC1CNC(c1cc(C(C)(C)C)no1)=O)=C(C)C C#CC1(O)CCN(C(C)C(=O)NCCC2CC(Nc3snc(Cl)c3C#N)C2)CC1 Cc1ncncc1C(N1CC2C(CN(C(=O)C(=CC3CCCCC3)F)C)C2C1)=O C(=O)(CCP(C)(C)=O)N1CCC(c2ccccc2)(NC(C)=O)C1 C1(C(=O)Nc2c(F)ccc(C)c2)C2CC(O)C(C2)N1C(C1COC(C)C1)=O N1(C(c2n[nH]c(CC)c2C)=O)CCN(C(C2CC2C2CC2)=O)CC1CCO C1(OCCS(=O)(=O)NCC(C)(C)N2CCCC2)CCCCC1 c1(C(N2C(CN(C)C)COCC2)C(=O)NC2CC(F)(F)C2)ccc2c(c1)OCC2 N1(C(COCC)=O)CCCC(CNC(C2(c3cccs3)CCCC2)=O)CC1 c1(C(=O)NCC2CN(C(C3CC3C(F)(F)F)=O)CC2O)cc2ccc(F)cc2o1 C1(F)(C(N(C)CC2N(C(C(CCSC)OC)=O)CCCC2)=O)CCCN(C)C1 C1(NC(C(CC)n2cncn2)=O)CN(C(=O)Cc2nc(C)no2)CC1OC C=CC1(C(=O)NCc2ncsc2C)CCN(C(c2cccc(F)c2)=O)C1 C1(COC(C(COCC=C)c2ccccc2)=O)CCC2COCCC2O1 N1(C(C(C)OCC=C)=O)CCC(CC)(NC(=O)C(c2c(C)nn(C)c2C)C)CC1 c1(C(C(=O)NC(CC)C)N(C2CCCCCC2)CC)cnn(C(C)C)c1I N1(C(=O)OC(C)(C)C)CCCCC12CCN(C(CC(O)C(F)(F)F)=O)C2 C1(NC(C(n2c(C)cc(C)n2)C)=O)CC(C)CN(C(=O)CCOC(C)C)C1 c1(-n2cc(-c3c(N)ccc(F)c3)nn2)c(Cl)cc(C(F)(F)F)cc1Cl C(CCCCC(=O)N(C1CCCC1(C)O)C)N(C(Cc1nc(C)oc1)=O)C Cc1cccnc1CC1CCC(N)C1.c1(N2C(=O)C2)nccc(C(F)F)n1 Cc1cc(C)n2ncc(C(N3CC4CCC(C3)C4N3CCCC(F)CC3)=O)c2n1 c1(C(=O)NCCC2CCN(C(C(C(C)OC)O)=O)CC2)cc(C)nc(C)n1 c1(C2(C(N3C(CNC(C(C)OCCCC)=O)CCC3)=O)CC2)ccccc1Cl N1(CCC)CCC(N=c2[nH]c(N3CCOC(CC)C3)nc3cccnc23)C1 CC(C)C(N=[N+]=[N-])C(=O)NCC(C)CNC(C1CCCN1C)=O N1(C(c2cn(C(CC)CC)nc2C)C(=O)NC2CC2)CCCC2(CNC(=O)O2)C1 C1(CCNC(C(C)(C)NC(=O)OC)=O)CN(C(=O)CS(C)(=O)=O)CC1C CC(CC(=O)NCC(CO)NC(=O)C1=CCCS1)C(F)(F)F C(=O)(C(C(C)(C)C)n1ccnn1)NCC(C)CNC(c1csnn1)=O O=C(C1CCCc2ccnn21)NC1CN(C(=O)C=CCF)CC12CCOCC2 N1(C(C=CC=CC)=O)CCC=C(C(=O)NCC2CC(O)C2(C)C)C1 N1(c2ccc(C(N)=O)nn2)CCCC2CCC(F)(F)CC12 C=CC(CC)C(=O)N1CCC(CO)(CNC(c2cnc(CC)nc2)=O)C1 N1(C(C2(CC)CCCO2)=O)CCCC(CCNC(=O)CN2CCCCCC2)CC1 C(=O)(C(CNC(=O)Cc1cc(C)n(C)n1)C(C)C)NCc1cc(C)sc1 C(CC(CC)C(=O)NCCCC(C)(C)NC(c1ncccc1Cl)=O)=CC C1(C(N(C)CC2(O)CN(C(C3CCC(CC)O3)=O)C2)=O)CCc2n[nH]cc2C1 C=CCCC(CC(C)C)C(=O)NCC1CN(C(c2ccnc(OC)n2)=O)CCO1 C12(C(=O)NC(CNC(C3(CC)CCC3)=O)CC(C)C)CC(C1)S(=O)(=O)C2 c1(C(=O)NCCCN(C(C2C(=C)CC2)=O)C2CC2)cnc(C)nc1C c1(OCCOC)ccccc1C(=O)NCCCCC1CN(C(=O)C2=CCCC2)C1 C1(CNC(CC(C)(C)F)=O)CN(C(=O)C(CO)N(C)C)CCC12CCOCC2 c1(CCNC(N2CCCC(OC)C2)=O)cnn2c1CCCC2 CC1CN(C(=O)CCc2cscn2)CC1NC(=O)CCCNC(=O)C(C)(C)C c1(C(=O)NCC(CN(C(C(C(C)C)OCC)=O)C)O)c(Cl)ccc(F)c1C CCC(C)CC(C(=O)N1CCCOC(C)(C)C1)NC(=O)Cc1cc(C)n(C)n1 C(=O)(C1CCc2nccn21)NCCC1(NC(c2cccc(C(C)C)c2N)=O)CC1 C(=O)(C(O)C(C)(C)CC)NCC(CNC(c1c(CC)ocn1)=O)F c1(CC)ncsc1C(=O)NC(C(=O)N1CC(CS(C)=O)C1)C1(O)CCC1 c1(C(N2CC(NC(CN(C)CC)=O)C(OC)C2)=O)ccn2cc(C)nc2c1 C1(NC(=O)Cc2ccccn2)CCC2(CC1)CC2NC(C1CCC(C2CC2)O1)=O N1(C(C2CC(CC)(CC)C2)=O)CC(NC(=O)C(C)N(C)C)C2(CCC2)C1 C1(NC(CCCC(=O)N(C)C)=O)CCN(C(C2CCC3(CC2)CC3)=O)CC(O)C1 c1(NC(C2CCCN(c3c(C)cnc(C)n3)C2)=O)nc(C)n(C)c1C#N N1(C(C(C)NC=O)=O)CC(C2CC2C(=O)Nc2ccccc2OCC2CC2)C1 CP(C)(=O)c1cc(NC(c2ccccc2-c2ccc3occc3c2)=O)ccn1 c1(C(N2CC(F)(CNC(C3C=CCS3)=O)C2)=O)cc(Br)ccn1 N1(S(C(C)C)(=O)=O)CCC2(CCN(C(=O)Nc3ccc(F)c(F)c3)C2)C1 Cn1cc(S(=O)(=O)NCC(=O)NCC(O)CNC(c2ccncc2F)=O)cn1 C(CCC(C)C)(C(=O)N1CCC1)NC(c1cncc(NC)c1)=O CC(C)(C)CC(F)C(=O)N1CCC(F)(CNC(=O)COCc2nccs2)C1 C(=O)(CCCCc1cn(CCCC(=O)O)nn1)N(C)CC1CC(C)C1 C1(OC)CN(C(c2c[nH]nc2C2CCCO2)=O)CC1NC(=O)CSC(C)(C)C N1(C(c2cccn3ccnc23)=O)CCCC2(C1)OCC(O)C2O N1(C(=O)NCC(C)(C)OCC)CCC(Oc2ccc(OC)cc2)CC1 C(=O)(C(C(C)(C)C)N(C)C)N(CC(CC)NC(C1CC(F)C(=O)N1)=O)CC C(=O)(CC(C)(C)C(F)(F)F)Nc1occ(C(C)(C)C)n1 c1(C(C(=O)NCCN(C(C2CCC(C)O2)=O)C)C)ccc(Cl)c(Cl)c1 c1(O)ccc2c(c1)CCC2.N1(C(=O)COC)CC2(CNC(=O)C3CC3)CCC1CC2 O=C(C#CC1CCCCO1)NCCC1(O)CN(C(=O)C2=COCCC2)C1 c1(NCC(N2CCCC2)C)cc(=NC(C)CCCO)[nH]c(C(C)C)n1.CCO CCC(CC(=O)NCCN(C(=O)C(CC1CC1)OC)C1CCCC1)C(C)C c1(C(N2CCC(CNC(C3(C(N)=O)CC3)=O)C(O)C2)=O)cccc2c1OCC2 n1(CCOC)nnnc1C(C(C)CC1CCCCC1)NC1CCOC1 c1(C(=O)NC2CCCCC2CNC(C2CC2(F)F)=O)ccc2ccncc2c1 c1(C(=O)NC2(CC=C)CN(C(=O)CCC(=O)OC)C2)cc(OC)cc2c1CCC2 Cc1cc(C)c(C(=O)N(CCCCN(C(=O)C(C(C)C)NC(N)=O)C)C)c(O)n1 N1(C(CC=C(C)C)=O)CCCCCC(NC(=O)C(C)(C)c2ccsc2)C1 Cc1cc(-c2cn(CCNC(c3cnc(C(F)F)nc3)=O)nn2)cnc1C C1(C2(O)CCC2)(C(=O)NCC2(CNC(C3(C4(C)CC4)CC3)=O)CC2)CC1 CC(N=c1[nH]c2c(c(=NCc3ccn(C)n3)[nH]1)COC2)c1ccc2ncsc2c1 c1(NCC(C(C)C)(C)NC(C2CC=CCO2)=O)cc(C(F)(F)F)nc2ncnn12 C(C(CC)(CC)C(=O)NC1CN(CC(F)F)C1)NC(COCC(=C)C)=O CC1CN(C(=O)CC(F)F)CCC1NC(=O)C1=COCC1 c1(C(N(CC(CNC(C2C(C=C)OCC2)=O)O)C)=O)ccc2cn(C)nc2c1 C1(c2n(C(CC)C)nnn2)(NC2CC(NC(=O)OCC)C2)CC2(CCNC2=O)C1 N(C1CCNc2ccc(C(=O)O)cc21)S(Cc1cc(OC)ns1)(=O)=O Cc1cc(=NCCC2C(C)CCCN2C(c2cccnn2)=O)c(C#N)c[nH]1 C(CCF)(C(=O)N1Cc2ccccc2CO1)NC(C1CC(CF)C1)=O c1(CC(C(=O)N(C2CCN(C(=O)C3=CCSC3)CC2)CCC)O)cccc(Cl)c1 N1(C(C(C)(C)OC(C)C)=O)CCC(CF)(NC(=O)Cc2cncn2C)C1 C1(CCOC)(C(=O)NCCCNC(c2ccnn2CCF)=O)CCNC1=O C1(C(N2C(C)CC(NC(=O)Cn3cc(C#N)cn3)CC2)=O)CCC2(CCCC2)C1 N1(C(C)=O)CC(O)CC1C(=O)N(C)CC1CCCN(C(=O)COCP(C)(C)=O)C1 C1(NC(C(CCC#C)O)=O)C2CC3CN(C(c4ccc(C)c(C)c4N)=O)C1C3C2 N1(C(C2C(SC)CN(C(=O)CCC3CCC(=O)C3)C2)=O)CC2CCC=CC12 C1(F)(C(=O)NC2CC(C)(NC(C(C)Oc3ccc(Cl)cc3)=O)C2)CCS(=O)(=O)C1 C(=O)(C(CCN(C)C)NC(=O)CC1CC1)NC(CC(=O)OCC)C C1(NC(c2ncc(C)cc2F)=O)CC2CCC(C1)N2C(C1CCOCC1)=O c1(CC)cnn2ccc(C(=O)N(C(C)CCNC(=O)C(C(C)C)N(C)C)C)nc12 C=CC1OCCC1NC(c1c(F)cncc1Br)c1nnnn1CCCC C1(c2n(CC=C)nnn2)(NCCc2ccc(Cl)s2)CCOCC1 C1(NC(C#CC(C)(C)C)=O)CCC2CN(C(=O)C=C3CN4CCC3CC4)CC12 CC(C1COc2ccccc21)NC1(c2nnnn2C(C)(C)C)CCC1C1CCC1 C12(C(=O)NCC(C(=O)Nc3ccc(OC)nc3)(C)OC)C(=O)C3CC1C2C3 c1(C(=O)NC(CNC(CCC(=O)OCC)=O)CO)c(Br)nc2n1CCC2 Cc1[nH]c(C(=O)Nc2ccc(C3CC3)nc2)c(C)c1C(N1CCCC1)=O C12(C(N3C(C(=O)OC)CC3C)=O)CCN(C(=O)C=CC(F)F)CCC1C2 N1(C(CN(C)C2CC2)=O)CCC(NC(C2CC2(Cl)Cl)=O)CC(C)(C)C1 C(=O)(C(C(C)C)NC(C1(F)CN(C(C2CC(N(C)C)C2)=O)C1)=O)OC c1(C(N(CC(C(=O)N(CC(O)CO)C(C)C)C)C)=O)cc2cccnc2[nH]1 c1(C(N2C(CC(N3CCC(C(=O)OCC)C3)=O)CCC2)=O)ccc(Cl)c(OC)c1 C1(C(N2CC(n3c(C)ccn3)C2)=O)CC(=O)N(c2ccccc2F)C1 Cc1cc(NC(=O)NC(C)CNS(C)(=O)=O)cs1 C1(CNC(NNC(c2ccc(N)cn2)=O)=O)CCC(C2CC2)C1 C(=O)(C1=CC2CCCC12)NCCCC(C)(C)NC(=O)COc1cccc(Cl)c1 c1(CNC(c2c(NCc3c(C)csc3)c[nH]n2)=O)n[nH]c2ccc(Br)cc12 c1(OCC#C)cccc(NCC2CCOC2)c1 Cc1nnc2n1CC(C(=O)NCC1CCCCC1NC(C1CNC(=O)N1)=O)CC2 c1(OC)ccc(C)c(CNC(=O)NC2CCN(c3ccccc3C(C)C)C2=O)c1 c1(C(N2CCN(c3ncc[nH]3)CC2)C(=O)NCC)cc(OC)c(O)c(Br)c1 CC(C)C#CC(=O)N1CCC1CNC(=O)Cn1nnnc1-c1ccsc1 C1(NC(c2c(NC)cccc2)=O)CCN(C(c2ccc(OC)cc2C)=O)CC1C Cc1cccn2ncc(C(N3CC(CNC(C4CCCC(=O)O4)=O)C(O)C3)=O)c12 c1(-c2cc(OC)ns2)ccc([N+](=O)[O-])cc1.C1(CCc2ccsc2)C(=O)OCCN1 C1(CN(C(=O)NC(c2ccsc2)CC)C)CCCS1 c1(CC(=O)NC(C)CCN(C)C(C2(CO)CCC2)=O)ccc2n[nH]cc2c1 C(CC(O)C(=O)N1CCC(CNC(C=CC(C)(C)SC)=O)(CO)C1)SC Cc1cc(C(N2CC(CNC(=O)CC3CCOCC3)C(O)C2)=O)cc2nc[nH]c12 Cc1ccc(C(C)(C)C(=O)NC2(CNC(=O)CSCC(C)C)CCC2)cc1 C(CCCN=C(NCC1CC2(CCOCC2)C1)NC1CC1)OCC C#CC1CN(C(c2cccnc2)=O)CCN1C(C1CC1F)=O S(=O)(=O)(c1ccc(Br)c(C#N)c1)Nc1cc(C)cc(C(=O)OCC)c1O CCC(CC)C(=O)NC1CCCC1C.O(CP(C)(C)=O)C(=O)C CC1CCC(NC(=O)C(N2CC(O)(CNC(C3CC4(CC4)C3)=O)C2)=O)CC1 C#CC1CN(C(c2cc(CC(C)C)on2)=O)CCN1C(c1ncn(C(C)C)n1)=O C(=O)(C1=CCCCC1)NC1C(CN(C(CC(=O)OCC)=O)C)CCC1 N1(C(c2n(C)ncc2Cl)=O)CC(C(N2CCCC2)=O)CCC1(C)C N1(C(c2c(C(C)C)snn2)=O)CC2OCC(NC(c3ccccn3)=O)C2C1 CC1(C)CC(C)(C(=O)NC(C2CCN(C(c3ccccc3C3CC3)=O)C2)(C)C)C1 C1(C)(CC(=O)NCC(CN(C)C(c2cnc(C(C)(C)C)[nH]2)=O)O)CC1(F)F C(=O)(C1COc2ccccc21)N1CCC(N(CC#C)C(C2CCS2(=O)=O)=O)CC1 C12(C(=O)NCCCN(C(C3(C)CC3)=O)CC3CCCC3)CCC(CC1=O)C2(C)C C1(CNC(CC(C)C)=O)CN(C(=O)C(C)(C)N2CCCC2)CCC1C c12ncc(C)cc1S(=O)(=O)NC1(CC1)CN2.c1(CC)ocnc1C(F)F c1(NC(C2C3(CCN(C(C4=C(C)OCC4)=O)C3)C2)=O)cc(I)cc2[nH]ccc12 c1(C(=O)NC(CN(C(c2cc(C)c(Cl)s2)=O)C)C)ccc2c(c1)CN(C)C2 N1(C(C(F)=C(C)C)=O)CCC(C(N2CCCCC2CF)=O)C12CC2 C1(NC(COCC(=O)NC)=O)(CNC(=O)CC2COCCO2)CCOC1 N1(C(C(CC=C)(C)C)=O)CC2CCCC2(CNC(=O)C2=NNC(=O)CC2)C1 C(=O)(CC=CCNC(=O)CCNC(C1CCCC1)=O)OCC c1(NC(C(CNC(CCn2ncc(C)c2)=O)(C)C)=O)ccc(C#N)cc1O C1(NC(=O)OC(C)(C)C)CC(O)CN(Cc2ccn(C3CC3)n2)C1 N1(c2cc(NCc3cc(C)nn3C)nc(C)n2)CCc2cc(F)cc(F)c2C1 C(C)(CC(C)N=c1[nH]c(Cl)nc2c(F)cc(C)cc12)c1cc(C)c(Br)c(C)c1 N1(C(C=CSC)=O)CCCCC(Nc2cc(C(C)C)ncn2)C1 c1(C(N(C2CCN(C(C(C)CC(C)(C)C)=O)CC2)C)=O)cc2cc(F)ccc2o1 c1(C(COC(C2CC2Cl)=O)=O)sc2ccccc2c1Cl C1(C(=O)NCC2(C)CCN(C(C3(F)CCCCC3)=O)C2)SC2C=CC1CC2 Cc1c(C(=O)NCC2CN(C(c3cn(C)nc3O)=O)CCO2)[nH]c2ccccc12 C(CCCCN(C)C(C1CCCS1)=O)NC(C1C(C)C1C)=O c1(C(=O)NC2C(OC)CN(C(=O)CCc3cccs3)C2)c(C)sc(C)c1C#N CC(CNC(c1cc2n(n1)CCC2)=O)C(F)C(=O)Nc1cc(CO)cc(F)c1 C1(CC(=O)N(CCO)CC)CCCN(C(c2cn(C)nc2COC)=O)CC1 C(=O)(NN1CCCC1C(=O)NC(C(O)CO)C1CC1)C1(C=C)CCOCC1 c1(CC(=O)NC2CCN(c3snc(COC)n3)C(C)C2)ccc2ncccc2c1 C12(NC(C=CCOC)=O)CCCC1N(C(c1cc(F)c(Cl)cc1F)=O)CC2 C1(NC(c2cnccc2Cl)=O)CC2CCC(C1)N2C(=O)C=CC1CCCC1 C1(CN(C)C(C2COCCO2)=O)CCN(C(=O)NC2CC2)C1 C1(CN(C(C2(C#C)CC2)=O)C)CCCN1C(c1cnccn1)=O c1(CNC(COCC=C)=O)ccc(C2CCOC2)cc1.C12(CCC1)C(=O)N(C)C2 S(=O)(=O)(c1cc(C(=O)NC2CCCC(NC(C3(N(C)C)CC3)=O)C2)co1)NC C1(C(=O)NCC(C2CC2)SC)C2CCN(C(C3CCCC3F)=O)CC12 c1(CN(C(C2CCC(C)CC2)C(=O)NC2COC2)C)cncc2ccccc12 C1(C2CCCCC2)(NC(C(CC2CC2)NC(C2C(C)(C)CCCO2)=O)=O)CC1 CC1CCN(C(C2Cc3cscc3C2)=O)C(C)C1NC(=O)C=CCN(C)C c1(OC)cccc(F)c1CC(N1CC2CC1CN2C(c1ccc(O)cc1F)=O)=O Cc1c(C(N2CCC(C(O)CNC(=O)C(O)c3ccco3)CC2)=O)[nH]ccc1=O N1(C(CSCC(C)C)=O)CCN(CCCO)CC1C.C1(=O)C(C)OCCN1 c1(C(=O)OC)ccnc2c1CCC2NC(c1cccc(C)c1C)=O C1(NC(CSCC)=O)CN(C(c2ccc(C3CCC3(C)C)cc2)=O)CC1(C)C C(=O)(CCCCCC)NC(C(CO)NC(CCNS(CC)(=O)=O)=O)C c1(C(N(CCN(CC=C)C)CC)=O)conc1CNC(=O)C=CCN(C)C CCCCCC(C)CC(=O)N(C1CCN(C(=O)C(CC)(CC)CO)CC1)CCO CC1=C(C(=O)NC(CCF)C(=O)NCC(C)(C)CN(C)C)CCO1 c1(-c2c(C(N3CCC(C(F)(F)F)C3)C)csc2)ccc(CN2CCCC2)cc1 N1(C(C)=O)CCC(C)(C)CC1N(CC1=NOC2(CCC2)C1)C(=O)C(N)=O c1(CC(=O)N(CCN(C(C(CC)=CCCC)=O)C)C)nc2ccccc2s1 C1(C(C)(C)C)CN(CCOC2CCS(=O)(=O)CC2)CCC1O c1(C(=O)NCc2c(CNC(=O)OC(C)(C)C)nccc2)ccc2c(c1)OCO2 C1(NC(C(C)=CC2CC2)=O)CCCC12CN(C(C1COC(=O)N1)=O)C2 C1(CC(C)O)CCN(C(=O)NC(C23CCC(CC2)O3)C2CC2)CC1 CC1(C)CN(C(C2C(C#N)C2(C)C)=O)CCC1C(N1CC(OCCF)C1)=O N1(C(c2c(SC)ccs2)=O)CC2(CCC2NC(C2CC3C=CC2CC3)=O)C1 N1(C(c2c(C)coc2)=O)CCC2(CO)CN(C(C3CC4(C3)CC(C)C4)=O)CC2C1 C(=O)(CCCC(=O)NCc1nocc1C(N1CC2CCC2(C)C1)=O)N(C)C c1(C(=O)NC)cccc(SC)c1.C12CCC(C1)N(C)C2C(=O)NC(C)(C)C C1(C)(CC)C(=O)NCCN1C(c1cc(Cl)ccc1NCC(=O)OC(C)(C)C)=O N1(C(C(CCCCC)O)=O)CCC(NC(=O)Cc2ccnn2C)C2(CCC2)C1 C1(=CC(=O)N(CC(C)NC(=O)CSc2nccn2C)C)CCC(C)(C)CC1 Cc1ccc(C(=O)NC2CCCC2CNC(c2coc(O)n2)=O)c(Br)c1F N1(C(CC(CNC(c2c[nH]c(C(N)=O)c2)=O)OC)=O)CC(O)(C2CCC2)C1 N1(CC)CCC(CNC(C2(C(C)C)CCN(C(c3cnc[nH]c3=N)=O)C2)=O)CC1 C(C(CO)(CO)NC(=O)CC(C)SC)N(C(c1nc(OCC)oc1)=O)C C1(CC(=O)NCCCCCNC(C2(C)CC2C(F)F)=O)C2CC3CC(C2)CC1C3 C(=O)(CCCCN(C(=O)CCCNC(N)=O)C)NCC1(OC)CCC1 c1(C(=O)NC2C(NC(Cn3ncc(P(C)(C)=O)c3)=O)C2)c(F)ccc2occc12 CCC1=NOC(CC(=O)NCC2(F)CC(C(=O)NC3CCC4(CC4)C3)C2)C1 N1(C(C(CC=CC)C)=O)CC(NC(c2c(C)nn(C(C)(C)C)c2C)=O)CC(F)C1 C1(CCOC(c2ccc(-c3nnco3)cc2)=O)COc2ccccc2O1 c1(C(N2C3C(NC(C(C4CCCC4)OC)=O)C(C3)C2)=O)ncc(F)cc1F c1(C(=O)NC(CC)(CC)CCNC(=O)CN2CC=CC2)cc(C)cn2ccnc12 CC(C)C(C)(C)C(=O)NCC1CCCCC1NC(c1cc(Br)sn1)=O N1(C(CN2CC(=O)NC2=O)=O)CC(NC(=O)Cc2cnns2)C2(CCC2)C1 CCCN=C(NC1CC1COC)N1CCC(S(=O)(=O)N2CCCC2)C1 Cc1nc(C(=O)NCC(C(C)C)NC(C2CCN(CC(C)C)CC2)=O)cc(O)n1 c1(NC2CCC(CC)C2)ccc2sc(C(=O)OC)cc2c1Br c1(C(N2C(CO)CC(NC(C3(C)CC=CCC3)=O)C2)=O)cc2n(n1)CCO2 S(=O)(=O)(c1ccccc1F)Oc1cncc(C(N2CCN(C)CC2)=O)c1 N1(C(C(C)NC(=O)NC)=O)CC(NC(=O)C=C(C)C2CC2)C(C)(C)C1 O=C(N=c1[nH]sc2ncccc12)C1C2CC1N(C(=O)Nc1cccc(Cl)c1)C2 C(N=c1nc2sccc2c(N2CC34CCC3(COC4)C2)[nH]1)C1C(CC)C1 c1(NC(c2c(COC)cc[nH]2)=O)ccc(NC(=O)C(=Cc2c[nH]cn2)F)c(C)c1 C(C(CNC(c1cccc(Cl)c1Cl)=O)C(F)(F)F)NC(C(C)SCC)=O c1(C(N2C(C(=O)NCc3nn[nH]c3C3CC3)C3CC3C2)=O)cccc2c[nH]nc12 C1(O)(NC(C(CC2CCCC2)NC(C(N2CCOCC2)C)=O)=O)CCOCC1 c1(C(=O)NC(C)C(C)C(=O)N2CC(F)C2)cccc2ccnn12 C1(C(=O)NC(C2(C(=O)NC(c3ncc(C)o3)C)CC2)C)CC12CCOC2 c1(C(N2CC(CCNC(CC(C=C)C)=O)OCC2)=O)ncc(CC)cc1C C=CCCC(=O)NCC=CCNC(=O)CC(=O)OCCOC c1(N2C(CC(C)NC(=O)C(C3CCC(=O)N3)C)CCC2)nc2cc(Br)cnc2s1 CCC(CC)CCCC(=O)N1CC2CCC(NC(c3ccc(OC)cc3)=O)(C2)C1 N1(C(C(C)NC(C)=O)=O)CC(NC(c2ccc(C(C)C)c(Cl)c2)=O)C2CC2C1 Cc1cc(C)c(CC(=O)NCCC2CN(C(c3cc[nH]n3)=O)CC2C)s1 c1(NCc2cn(CCNC(C3C(C)CC(=O)CC3)=O)nn2)ccc2ccncc2c1 c1(C(C)=O)c(C)[nH]c(C(=O)Nc2ccccc2OC2CCOC2)c1C(C)C C1(CNC(C)(C)CN2CCCC2)C2CC1N(C(=O)OC(C)(C)C)C2.C(=O)C(C)(C)F N1(C(C(c2cccnc2)NC(C2CCC2(F)F)=O)=O)CC(F)(F)C1C1CC1 C1(NC(=O)Cc2ccccc2)COC2(CNC(C3CC4(C3)CC(O)C4)=O)CC1C2 C1(C(=O)NC2CC(C(N(C)Cc3c(C)nsc3)=O)C2(C)C)CCC(O)CN1C Cc1cc(C)n(CC(N2CCN(C(c3cnc(O)n3C)=O)C3CC23)=O)c(=O)n1 CCCCCC(CCCCC)CC(=O)N(CC(O)CNC(C1CC1COC)=O)C Fc1cc(Br)c2nccc(N3CCCC4NCCCCC34)c2c1 C1(C(=O)NCCCN(CC(=O)NCCCC)CC)(CC)CCOCC1 C1(C2(O)CN(C(=O)C(N3CCCCCC3)C)C2)(CNC(CC(C(C)C)C)=O)CC1 N1(C(C=CC(CC)C)=O)CC(NC(=O)CN2CCCCC2C)C(N=[N+]=[N-])C1 N1(C(c2cc(CCC)nn2C)=O)CCN(C(C2(Cl)CC2(F)F)=O)CC(O)C1 Cc1ncoc1C(=O)NCC1CCCC1NC(C1CN(S(C)(=O)=O)C1)=O C(=O)(C(C)CCCC)N(C)CC1N(C(CSCC#C)=O)CC(F)C1 c1(C(=O)NC2CCCC(CN(C(=O)C(F)(F)CO)C)C2)cc2cn[nH]c2cn1 c1(C(=O)NC2(CO)CCN(C(C3CC4CCCCC34)=O)C2)cncc2c1CCC2 C1(OCC)CC2(CCC2)C1OC1CC(c2ccccc2)(CC)C1.C12CN(C1)C(=O)N2 C1(CCC(=O)N(C)CCNC(C2(C(N)=O)CC2)=O)CCC(=O)C1 C1(C(C)NC(c2c(CC)nn[nH]2)=O)CCN(C(c2cn(CC3CC3)nn2)=O)CC1 C1(COCC)CCCCN1C(c1cnc(CNC(c2nccn2C)=O)nc1)=O N1(C(C2=CCCN(C(=O)CC3COCCO3)C2)=O)CC2CSCC(C2)C1 N1(CC(N2CCN(C(C(CC)(C)O)=O)CC2)=O)OC(C)(C)CC1=O Cc1cc(C(=O)NCCC2(O)CN(C(C3CC3C3CCCC3)=O)C2)ccc1Cl c1(C(=O)NC(CCN(C(C(CC)CC)=O)C)C(C)C)cc2c(C)c(Cl)ccc2[nH]1 N1(C(CN2CC(CSCC)C2)=O)CCN(C(c2ccc(C(=O)OC)cc2)=O)CC1 Cc1cc(C(=O)NCCC(C)NC(c2ccsc2C(F)(F)F)=O)c2[nH]cnc2c1 C(CCCCC(=O)N(C)CCN(C(c1cncc(C2CC2)c1)=O)C(C)C)NC(C)=O C1(NC(C(C=CC)O)=O)CCCCN(C(=O)Cc2cc(C)ccc2OC)C1 c1(C(N(C(C)C(=O)Nc2cnc(OC)nc2)CC)=O)cccc(C#N)c1 CC1SCCC1C(=O)Nc1ccsn1.C1(=O)CCCC2(CCC2)N1 N1(C(CCCC=C)=O)CCC(NC(=O)CCOC)CC(C)(C)C1 c1(NC(C)C)cc(NC2CCN(CCc3ncnn3C)CC2)nc(C(F)(F)F)n1 N1(C(c2c(CNC(C3CC=CCC3)=O)n[nH]c2)=O)CCCC2(CCOC2)C1 CC(=O)CCCC(=O)NCC1CC(C)(C)CN1C(=O)Cn1cnc(C#N)n1 c1(-n2cc(C3CN(C(C4CCSC4)=O)C3)nn2)cc(F)ccc1Cl c1(C(=O)NC(CC(C)NC(=O)CCc2cccs2)C)cc2c(cc1Cl)NCC2 C(=O)(C1=CCC(NC(c2cc(Cl)cs2)=O)C1)NC(c1nnc(C)o1)C CCCCCC(C)(CC)C(=O)N1CCN(C)C(CNC(C2(OC)CC2)=O)C1 c1(CC)ncc(C(=O)NC2(C)CN(C(c3cc(C(C)C)nn3CC)=O)C2)c(C)n1 Cc1c(F)ccc(C(=O)NCC2(NC(=O)C=CC3CCCCC3)CCC2)c1Cl N1(C(COC(=O)C(C)OCC(F)(F)F)=O)CC(NCc2onc(C)n2)CC12CCC2 c1(OC)ncnc(OC)c1NC(C1(C)CCCN(Cc2cc(O)ccc2C)C1)=O C1(N(C)C(C2(F)CCCOC2)=O)CCN(C(=O)Cn2ccccc2=O)CC1 c1(C(=O)NCC2C(C)CN(C(c3cccs3)=O)C2)n[nH]c2c1CCC2 C(CC(C(=O)NCc1nnc(CC)o1)NC(c1ocnc1CC)=O)OCC C1(C(N(C)Cc2n(CC)ccn2)=O)CC2CCCC2N1C(C1CC=CC(O)C1)=O C1(NC(C=CC(CC)C)=O)CN(C(c2cc(Cl)cn2C)=O)CCC1CO C1(C(N2C(C(N(C)Cc3c(C)occ3)=O)CCC2)=O)CC2C(C1)C2(F)F N1(C(C(CCC)O)=O)CCC2(CCCN2C(C2(c3ccc(Br)cn3)CC2)=O)C1 c1(OC)cc(C)c(C)cc1S(=O)(=O)CNC(=O)C(=O)NCC1CCC1.c1ccccc1 CN(CCCC(=O)NC1CCC12CN(C(c1cc(C3CCCC3)no1)=O)C2)N=O C1(NC(c2c(C)ccs2)=O)COC2(CCCN(C(c3ccc(O)nc3)=O)C2)C1 c1(C(C(=O)NC2COC2)N(c2ccc(C)c(F)c2)C)cc(F)c(Cl)cc1Cl N1(C(c2c(=N)[nH][nH]c2)=O)CCC2(CC1)OCCC2NC(=O)Cc1cnco1 N1(C(C2C(CC(C)C)C2)=O)CC2(CCCCN2C(=O)Cc2coc(C(F)F)n2)C1 CCCC(CC)C(=O)NCC(C)N(C)C(c1cccc(CC#N)c1)=O N1(C(c2cc(C(=O)OCC)n(C)n2)=O)CC(C)N(C(c2n[nH]c(C)n2)=O)CC1C N1(C(=O)NCCC=C=C)CCOCC1c1noc(C(=O)OC)n1 N1(C(CCCC(C)=O)=O)CCC2(CCCN(C(C34CCCNC(=O)C3C4)=O)C2)C1 Cc1cc(C(=O)NC2(CNC(C3CCC3)=O)CCOCC2)ncc1CO Cc1cc(C(N2CC(CC(=O)NCCN3CC(C)(O)C3)C(C)C2)=O)cn1C Cn1ncc(C#N)c1C(=O)NC1CC(CC(N2CCC(CO)C(O)C2)=O)C1 C(=O)(C1=CCC(C)(C)CC1)N1CCOCC(NC(CCS(=O)(=O)N(C)C)=O)C1 C1(C(N2CC3CCC3C2)=O)CCS(=O)(=O)N1 C(=O)(CC(C)C(F)F)N(CCC(C)NC(c1cnn(C(C)C)c1Br)=O)C CC1CC(NC(=O)C=Cc2ccco2)CCN1C(c1ccc(F)cc1)=O C1(NC(c2cc(C)sn2)=O)CC(CNC(=O)CCN2CCCS2(=O)=O)C12CCC2 C(=O)(C(O)(C(F)(F)F)C1CC1)N(CCCn1cc(C(C)O)nn1)CC1CC1 c1(C(=O)OC)cc(NC(=O)NCCOC2CCCC(C)C2)c(Cl)c(C)c1 C1(CNC(CSCCC(C)C)=O)CN(C(=O)CNC=O)CC12CC2 c1(C(=O)NCC(=O)NCC(C)Cc2ccccn2)nc(=N)cc[nH]1 c1(CC(=O)NC(CC)(C)CNC(c2ccc(C)o2)=O)ccc2scc(C)c2c1 C1(C(=O)NC2(C)CN(C(C(C(C)(C)C)SC)=O)C2)CCc2ncccc2C1 N1(C(=O)C=C2CCOCC2)CCC2CN(C(c3cccnn3)=O)CCC2C1 c1(CC(C(=O)N(CCCNC(C(CC)NC(N)=O)=O)C2CC2)C)ccccc1C CC1CN(C(C2(C)CC3(CC3)C2)=O)CCC1CNC(=O)CS(=O)(=O)N(C)C C1(COC)(NC(=O)Cc2cc(C3CC3)on2)CCN(C(C2CC(=O)C2)=O)CC1 C1(C(N2C(C)(CNC(c3nc(OC)c(C)s3)=O)CCC2)=O)CCOCC1(C)C c1(C2(NC(=O)NCCSCCCO)CC2)ccc(F)cc1Cl N1(C(C(CC(C)C)O)=O)C2CCCC1CN(C(=O)C(C)CSC(F)(F)F)C2 c1(OC)ccc(NC(=O)C(=O)NCC2CN(C(c3conc3C)=O)CCO2)cc1 c1(C(=O)NC2CCCN(C(C3CCC3)=O)CC2F)n[nH]c2ccc(Br)cc12 C1(NC(Cn2ncc(CC)c2)=O)C2CCCN(c3ccnc(CO)n3)C2C1(C)C C1(CCC(=O)N(C(CC)C)C)CCC(NC(C2CCC(=O)C2)=O)C1 c1(C2(C(=O)NCC(C)N(C(CC(C)N(C)C)=O)C)CCCC2)cccc(Cl)c1F c1(C(=O)NC2C(NC(c3n(C=C)ncc3)=O)COCC2)cc2c(cn1)CCCC2 N1(C(COCCN(C)C)=O)CC(O)CC1CNC(c1nncn1C1CC1)=O N1(C(C(c2cn(C)nc2)O)=O)C2CCC1C(C(=O)NC1CCC3(CCC3)C1)C2 CCCCCC(C)(C)C(=O)NC1CN(C(=O)C(C)(CC)CC)CCC1CO c1(C(N2CCC(N(C(=O)CC3COCCO3)C)CC2)=O)cc2sccc2s1 c1(OC)cc(I)ccc1NC(=O)COC(=O)C(C)(C)c1nn[nH]n1 CC1CCC(NC(=O)OC(C)(C)C)CN1CC(c1ccccn1)=O C(C(CCC)C(=O)N(CC(C(C)C)OC)C)NC(c1n(C=C)nnc1)=O c1(C(N2CCC(C)(C(=O)Nc3cncc(C#N)n3)C2)=O)ccc([N+](=O)[O-])nc1 CCC(CC)(CC)C(=O)N1CCOC(C)(CNC(c2cccc(F)c2Cl)=O)C1 C12(C(=O)NC3(C4N(C(CS(N)(=O)=O)=O)CCC4)CC3)C3C4C1C1C2C3C41C(N)=O c1(CCC(=O)NCC(c2ccc(O)cc2)(C)O)ccccc1F CCCC(C(=O)NCc1cc(C)ns1)NC(C1CCC(=O)N1)=O N1(C(C(=O)NC(C(C)F)C)=O)CCC(C(C)(C)C)(C(=O)OC(C)(C)C)C1 c1(C(=O)NC(C2CCOC2)CNC(COCCC#C)=O)cnc(O)n(C)c1=O Cc1cccc2[nH]cc(C(=O)NCC(C)N(C)C(c3csc(Cl)c3Cl)=O)c12 C(CCOCCO)(C(=O)N1CCC(CC(F)F)C1)NC(c1c(N)snn1)=O c1(N2CCC(NC(c3csnn3)=O)C(F)C2)nc(O)c2c[nH]nc2n1 C(=O)(C(C)CC#N)NCC1C(C(N(CC(C2CC2)OC)C)=O)CCC1 Cc1cnc2cc(C(=O)NC3CC(C)(NC(=O)CC4CC5CC5C4)C3)nn2c1 CC1(C(N2CCN(CCCNC(c3nocc3C3CC3)=O)CC2)=O)CCCOC1 C1(N(C(CCN(C)CC)=O)CC)CN(C(=O)CCc2ccco2)CC12CCC2 c1(C(N2C(CCNC(C=NOC)=O)CCCC2)=O)cc(C)c(N)c(C)c1 C1(C)(C(=O)NCC2N(c3cc(C(C)=O)ncn3)CCCC2)CC(O)CN1C c1(OC)ccnc(C(=O)NCC2CCCCN2C(C2CC(C(C)C)C2)=O)c1 C=CC(C)CCNC(C1(N(C(=O)C=CC)C)CC1)=O N1(C(C(CCC)OC)C(=O)NC2COC2)CCC(O)C(O)(C(=O)OC)C1 c1(C(=O)NCC2(NC(C(C)CO)=O)CCCCC2C)ccc2nc(Cl)nn2c1 c1(CCNC(N2CCC(n3cccc3)CC2)=O)ccnc(Cl)c1F c1(C(N2C(CNC(COCCCC)=O)CCC2)=O)cncc(C2CC2)c1 N1(C(CC2(C)CC2F)=O)CC(O)(CCNC(c2cnn(-c3ccncc3)c2)=O)C1 c1(N(CC)CC)ccc(NC(C2CC(O)CN2Cc2ccnn2C(C)C)=O)cc1 N1(C(C)=O)CC2(CCC2NC(=O)C(S(C)(=O)=O)c2ccccc2)C1 c1(C(=O)NC2CC2NC(C2(O)CCC2)=O)cnc2c(c1)CCCO2 C1(C(=O)OCC)CN(Cc2cnc(O)c(Cl)c2)CC12CCCCCC2(F)F c1(OCC(=O)NCC(CN(C)C(C2CCC2C(F)F)=O)O)ccccc1F C#CCC(C)(CC)C(=O)NC1CCN(C(c2cnn(CC(C)C)c2C)=O)CC1 C1(C(=O)NCC)(Cc2cn(CC=C)nn2)CCCN1C(=O)C(O)CN1CCCC1 CN=c1[nH]c(=NCCC2CC2C)[nH]c(=NCCc2cc(F)ccc2F)[nH]1 c1(C(=O)NC2CC(C)(NC(c3ccoc3Br)=O)C2)cnc2c(c1)NC(=O)CO2 CC1CCC=C1C(=O)NC1CCN(C(=O)C=Cc2ccncc2)CC1CO S(=O)(=O)(c1ccccc1NNC(=O)NCCN(C)C)N1CCCC(COCC)C1 C1(C)(OC)CC(Nc2cc(SCc3ccccc3)n(C(C)(C)C)n2)C1(C)C c1(CNc2c(N(C)C)ncc(Br)c2)cc(Cl)cc(F)c1Cl C1(NC(c2ccc(COC)o2)=O)CN(C(=O)C(CO)NC(=O)C(F)(F)F)CC1C c1(C(=O)NCc2nc(CNC(C(C=CC)O)=O)sc2)cnc(OC)nc1C C(c1ccccc1C(F)(F)F)=CC(N1CCN(C(=O)C2=CCCCO2)C2CC12)=O N1(C(c2cnc(C(C)=O)s2)=O)CC(C)N(C(=O)CC2=CCCCC2)CC1C C(CNC(c1cccnc1S)=O)(CC(=O)NCc1nc(C)cs1)OC C1(CNC(C(CNC(c2scc(C)c2C)=O)OC)=O)NC(=O)CC1(C)C C(C(C(=O)N1CCC1(C)C(N)=O)NC(=O)C(O)Cn1cncn1)OC(C)C C1(C(CNC(C(C)OCC=C)=O)(C)O)CCCN(C(=O)Cn2ncnn2)C1 c1(C(=O)NC(C(C)NC(Cc2cc(C)sc2)=O)C(C)C)cc(Cl)cnc1O Cc1ccc(I)cc1C(N1CC2CC1CN2C(=O)Cn1ccncc1=O)=O N1(C(c2ccc(N(C)C)cc2F)=O)CC(C2CC2(F)F)C1 N1(C(c2ccc(F)c(Br)c2)=O)CC2CN(S(=O)(=O)CC3CC3)CC2C1 C(CC1=CCCCC1)NC(C1C2CC3C(C2NC(C2COCOC2)=O)C13)=O n1(CC#C)cnnc1C(=O)NC1CCCC1CNC(C1CCCN1C(C)=O)=O Cc1cccc(Cl)c1OCC(=O)N(CCCCCNC(=O)C=C1CC1)C C#Cc1cccc(C(=O)NCCCCC(C)NC(C2CC2C)=O)c1C C(=O)(C#CC1CCOC1)N1CCN(C(c2cc(C)c(C)s2)=O)CC1C N1(C(C(N2CCCCCC2)C)=O)CCC(N(C(=O)C(C)C2CCCO2)CCO)CC1 C1(C)(C(=O)NC(CC2CN(C(CC(=C)Br)=O)C2)C)CCN(C)C1=O N1(C(CN(C)C(=O)C2CC2)=O)CCC(C)(NC(c2cc(Br)c[nH]2)=O)C1 N1(C(=O)C=CC2CCCN2C(c2cccc[n+]2[O-])=O)CCN2C(=O)OCC2C1 C(=O)(C1=CCCOC1)NC(CCNC(CN(C)CC)=O)C N1(CCCOCC)CCC2(CC1)COC(NC(=O)C(c1ccc(F)cc1)(F)F)C2 c1(C(=O)NCC2(COC)CN(C(CSCC#C)=O)C2)cnc2c(c1)COC2 N1(C(C(C)(C)NC(=O)NCc2ccc(C3CC3)o2)=O)CCc2ccccc2C1 CCCC(C)(CCC)C(=O)NCC1C=CCN1C(=O)Cn1cc([N+](=O)[O-])nc1C O=C(CCCC(F)(F)C(F)(F)F)NC1CC1c1ccn(CCOCCO)n1 C(=O)(N=c1nc[nH]n2c(Br)ccc12)N(C)Cc1cccc(C)c1 Cc1ccccc1CC(C)N(C)Cc1cnc2n1CCC2 C#Cc1ccc(Cl)c(C(=O)NCC(C)(C)CN(C)C(C2CC2CCC)=O)c1 N1(C(C2N(C(c3cc(C)nn3C(F)F)=O)CC2)=O)CCc2cnn(C)c2C1 C12(NC(C3COCCN3C(=O)C(F)n3ccnc3)=O)CCC(O)(CC1)CC2 c1(C(=O)NC2CCCC2NC(C2CCCCO2)=O)ncc(F)cc1F c1(C(=O)Nc2ccc(NCc3ccc(C)cc3)cn2)cc(F)c([N+](=O)[O-])cc1F Cc1ccc(C(N2CCC(NC(c3ncn(C)n3)=O)C(F)C2)=O)cc1[N+](=O)[O-] Cn1ccnc1CCC(=O)NC1CCC1CNC(=O)CC1CSCCS1 C=C(C(=O)N1CCN(C)CC1C(C)C)C1CCC(F)(F)CC1 N1(C(CC=CC=C)=O)CCC(=C)CC1C(=O)NC1CC2CC1CC2CO C1(C(N(CC)C)=O)CCCN(C(=O)CCNC2CCCO2)C1.C(C)=O c1(C(N(CCN(C(c2cnc(OC)nc2)=O)C)C)=O)cccc(C)c1N CC(C)CC(CC(C)C)C(=O)N1CC(C(C)NC(c2c[nH]ccc2=O)=O)C1 C1(CCNC(C=COCC)=O)CCCCN1C(c1cc(C)n(C2CC2)n1)=O Cn1cnc2c(C(N3CC4(CC4)CC3C(N3C4CCC3CC4)=O)=O)ncnc12 Cc1cn2c(n1)CC(C(=O)NCC1CC(O)CN1C(c1ncc[nH]c1=O)=O)C2 C1CCC(=O)N2CCC2C(=O)N1C.C1(C(=O)N(C)C)C=CCS1 C(C(O)CN=c1ccnc(C(F)(F)F)[nH]1)NC(C(c1ccc(F)cc1)C)=O Cc1cnc(C)c(NC(=O)CC2CC3(C2)CN(C(C2CCCCC2)=O)C3)c1 CS(=O)(=O)c1ccc(CN=c2nc(CCc3ccccc3)[nH]s2)cc1 C12(N(C)C(c3csc(Cl)c3)=O)CCCC1CN(C(=O)C=Cc1cnn(C)c1)CC2 N1(C(C(CC=C)NC(C)=O)=O)CCC(COC)(NC(=O)Cc2csc(=N)[nH]2)CC1 CC1(NC(C2CNC(=O)N2)=O)CC(NC(c2ccncn2)=O)C1 CON(CCC(=O)NC(CO)CCF)C(=O)c1cc(C(F)F)[nH]n1 N1(C(C(CCC)(F)F)=O)CCC(C(N2CC(C3CC3)(OC)C2)=O)CC1(C)C C(=O)(C1=CNC2=NCCCN12)NCC1N(C(CC(C=C)CC)=O)CCCC1 c1(C(=O)NCC2OCCCN(C(CSCC(C)C)=O)C2)csc2ccncc12 N1(C(CCN(CC)CC)=O)CC(CC(=O)NC2(CN3CCCCC3)CC2)C(C)C1 n1(CC)nc(C(N2CCC2CC(=O)NCC(F)Br)=O)c(C)n1 C(CCC(=O)N(CC(C)C(=O)NC1CCN(CC)C1)C)OCC=C c1(COC)nccc(=NC2CN(C(=O)CC3C=CCCC3)CC(C)(C)C2)[nH]1 C1(OC)CCN(C(C2CCN(C(=O)C3=COCC3)C2C(C)C)=O)C1C c1(OC)ccc(C(N2CC=CC2CNC(=O)C(n2cc(Cl)cn2)C)=O)nc1 C1(C)(C(=O)NCC(CC)n2cccn2)CC(O)CN1C(c1n[nH]c(=N)[nH]1)=O C1(NC(CC)CC2CCCCC2)CC12CCN(c1cc(OCCO)ncn1)CC2 C(C(CC(F)(F)F)NC(=O)C(O)c1ccco1)NC(C(C)(C)N(C)C)=O Cc1cn2c(n1)CC(C(=O)NCCC(C)NC(C1CCC(C(N)=O)CC1)=O)CC2 C(C(C)(CC(C)C)NC(=O)Cc1cc(C2CC2)no1)NC(CCC(C)OC)=O C1(C(=O)N(C)CCN(C(=O)CN2CCC(C)C2)C(C)C)(OC)CCOCC1 Nc1cc(C(N2CCCCC2CNC(=O)CC(C2CC2)C2CC2)=O)cc(Cl)n1 C1(CC(=O)NC2CCC2NC(=O)COc2ccc(C3CC3)cc2)COCCOC1 c1(SC)nc(=NC2CC(C)N(C(C3CCc4nnn(C)c4C3)=O)C2)s[nH]1 N1(C(C(C(C)NC(Cn2ncc(CC)c2)=O)(C)C)=O)CCOCC(C)(C)C1 N1(C(c2occ(OC)c(=O)c2)=O)CCCC2(NC(=O)CC3CCCC3)CC2C1 N1(C(C(C)C2CC2)=O)CCC2(CC1)CC(C)N(C(c1ccc(Cl)cc1)=O)C2 n1(C(CC)(C)C)nnnc1C(C(C1CCOCC1)C)NC1(CCF)CC1 Cn1cnc2cc(CN3CCNC(=O)C3(C)C)ccc12 N(C(=NCC(=O)NC(C)(C)C)NC1CCCSC1)C(C)Cc1ccccn1 C=C(C)C(C)(O)C(=O)NCCC(C)CCNC(=O)CCn1cnccc1=O CN1CCC(C(F)(F)F)(C(=O)NCC(C)(C)CCNC(=O)CNC(N)=O)C1 N1(C(c2ccn(CCC)n2)=O)CCC(C)CC1CNC(C12CCCC1C2(F)F)=O c1(CC)nc(C)c(C(N2CC(NC(=O)C=C3CCOCC3)C(C)C2)=O)o1 C(N=c1nc2c(c[nH]1)COCC2)C1(CCNC(C2C(C)(C(C)C)C2)=O)CC1 Cc1cccnc1C(N1CC(NC(=O)Cc2ccc(CN(C)C)cc2)C2CC12)=O C1(C(C)(C)C)CC(C(=O)NC2CCN(C(c3ccc(N)cc3O)=O)C2)=NO1 c1(CNC(C(CSC)OC)=O)cccc2c1OC(F)(F)O2 N1(C(c2nccc(C)n2)=O)CCC(NC(=O)Cn2ccc(C)cc2=O)CC1C c1(OC)ccc(O)cc1C(N1CCN(C(C2(C#N)CCCCC2)=O)CC1)=O c1(C(=O)NC2C(NC(c3c(SC)c(F)ccc3)=O)CC2)cnc2ccccc2c1 CCC(C(=O)N(C)C(c1c[nH]nc1COC(C)=O)=O)N(C)C(C1CC1C)=O c1(CN2CC(C)(CC(=O)NC(C3(C(=O)OCC)CCC3)=O)C2)cnnc(O)c1 C=CC(CCC)CC(=O)N1CCC(C)C(CC(=O)NCCCn2cncn2)C1 c1(N(C(=O)NCC2CC3CNC2C3)Cc2ccccc2)c[nH]c2cnccc12 c1(CC(=O)NC2C(CNC(C(C(C)C)OC)=O)CCO2)cccc(C#N)c1 c1(N(C)CC2CCN(C(=O)CN3C(=O)CCC3=O)C2)nc(Cl)ncc1C1CC1 C1(C)(C(=O)NCC(C)(C)CNC(C2CC(n3ccnn3)C2)=O)CCNC(=O)C1 C(CS(=O)(=O)CC(=O)OC1(C)CCS(=O)(=O)C1)NC(c1c(C)cccc1)CO CC(C)(O)CCC(=O)N1CC(CNC(c2cnc(C3CC3)s2)=O)C(C(F)(F)F)C1 N1(C(C2CC(OC(F)(F)F)C2)=O)CCN(C(c2cnns2)=O)C2COCC12 N1(C(C2CCS(=O)(=O)N2)=O)CC2CCCS(=O)(=O)C2C1 C(=O)(NN1CCCC(C(=O)O)C1)C1CCCC1.c1(CNC)cccc(F)c1 CC(C)(C)C(CNC(=O)CC(C)(O)C1CC1)NC(C1CC(c2ccccc2)C1)=O N1(C(C(C)C2CC2)=O)CCCCC(C2CN(C(C3CCC(F)(F)CC3)=O)C2)C1 CCC(CNC(C1CCC(NC(=O)C(F)CC2CCOC2)C1)=O)CO c1(C(=O)NC(C2(CNC(C3(OC)CCCC3)=O)CC2)C)ncnc(O)c1F c1(C(N2CCC(F)(CNC(C(CC)COC)=O)C2)=O)nc(C(C)C)ncc1Cl c1(C(=O)OC)cc(C)cnc1NC1CC(NC(=O)Cc2cc[nH]n2)C1 C12(NC(Cc3c(C(=O)OC)cccc3)=O)CCN(C(=O)CCC(C)C)CC1C2 S(=O)(=O)(c1cc(C)cs1)N1CC(C(=O)Nc2ccc(CCC)cc2)C(O)CC1 c1(CN2CC(NC(c3c(O)cc(O)cc3O)=O)C(F)(F)C2)cc(F)c(I)c(F)c1 N1(C(c2c(C)[nH]cc2)=O)CCN(CC(=O)NC(C)(CO)C2CCCC2)CC1 c1(C(N2CCC(NC(CCc3ccc(OC)nc3)=O)C2C)=O)cc2ccsc2s1 CCC(C(=O)NCc1ncoc1CCNC(=O)CN(CC(C)(C)C)C)C(C)O N1(C(CC(=O)OCC)=O)C2CCC1CC(CNC(=O)C1=C(Cl)CCC1)C2 c1(C(N2CCC(NC(=O)CCCn3cncn3)C2)=O)cccnc1Br N1(C(c2cnn(-c3ccccc3)c2)C(=O)NCC)CCC(O)(c2ccccc2)C1 C=CCCCCCC(=O)N1CCC(CF)(NC(c2cnc(-c3ccoc3)s2)=O)C1 Cc1nc(O)ccc1C(=O)NC1CCCCC1CNC(=O)C=Cc1cn[nH]c1 N1(C(CCCC#C)=O)CCN(C(C2CCN(C)C2=O)=O)CC12CCC2 C1(CC(N2CC(C)C(N=[N+]=[N-])C2)=O)CCCCC12NC(=O)NC2=O N1(C(C(C)CCO)=O)CCCC(NC(C2CCCC2C)=O)CC1 C(=O)(C#CC1CCCCC1)NCc1cc(C(N(CC#CC)CC#C)=O)no1 C1(F)(CNC(C(CC)n2ccnc2)=O)CCC(CNC(=O)Cc2ccon2)CC1 N1(C(CC)C)CCC(N=c2nc3scnc3c(NCc3coc(C)c3)[nH]2)CC1 c1(C(=O)NC2C(SC)CN(C(C3(C)CCCOC3)=O)C2)ccc2nnc(S)n2c1 N1(CCc2c(C(C)(C)C)cccc2)CCC(CNS(=O)(=O)CC2CC2)CC1 S(=O)(=O)(c1ccc(Cl)cc1)NCC1CN(Cc2c(OC)cc(F)cc2)C1 CCCC(C(=O)N(CCC(=O)NCC(=O)Nc1cccc(F)c1)C)N(C)C C1(c2cn(C)nc2)CC(c2nnnn2C2CC2)(NCCCOC(F)(F)F)CCO1 c1(CC(N2CCN(C(c3ncc(C)c(Cl)c3)=O)C3C2C3)=O)ccc2c(c1)CCC2 c1(OCC)cccnc1C(=O)NCCC1CC(NC(=O)C=C(Cl)Cl)C1 CC1CCC(CNC(=O)Cc2cnc(C3CC3)[nH]2)N(C(=O)C(=O)N=S(C)(C)=O)C1 C(c1cncc(F)c1)=CC(N1CC2C(NC(C(C(C)C)NC=O)=O)(C2)C1)=O c1(OC)cc(CC(=O)NC2CCCCC2CO)nc(OC)n1.C1(N)CSC1 N1(C(CC2(CSC)CC2)=O)CC2(C1)CN(C(C1CCS(=O)(=O)C1)=O)CC2CO Cc1cc(CC(=O)NCC(C)(F)CNC(=O)CN2C(=O)CCC2=O)ccc1O CCCC(C(=O)OC)C(=O)N1CCC(C)(C)C(NC(=O)Cn2cncn2)C1 C1(COC)CC(CNC(c2ccncc2F)=O)N(C(c2cnc(C(C)=O)s2)=O)C1 N1(C(C2(CCC)CCC2)=O)CC(CNC(c2ccc[n+]([O-])c2)=O)C(O)C1 N=c1[nH]c2c(s1)CCCC2C(=O)NC1CC(CNC(=O)CCc2cnn[nH]2)C1 C1(C(N2CCC(OCC(=O)NC(c3cccnc3)C)C2)=O)CCCN1C=O N1(C(COC(CNC(c2cncc(C=C)c2)=O)(C)C)=O)CCCC(C)(OC)CC1 N1(C(CC(C)(C)N(C(=O)CCCN=[N+]=[N-])C)=O)CCC2(CC1)CSC2 c1(NC(=O)C(c2ccc(Cl)cc2)=O)cccc(NC(c2cc(Cl)cs2)=O)c1 c1(C(=O)NC2CCCC(NC(c3c(C)cc(O)nc3)=O)C2)c(C)ccc(F)c1O c1(SCC)ccc(C(N2CCCC2CCNC(C2(C)CC2C)=O)=O)cc1 N1(C(CCn2c(C(C)C)ncc2)=O)CC(NC(c2ccncc2Cl)=O)C(C)(C)C1 C1(OC)CC(C(=O)NC2(C(C)(F)F)CC2)N(C(=O)C(C)CC#N)C1 c1(C(=O)NCCC(C)CCNC(=O)CC23CCCC2C3)cccc2nn(C)cc12 O=C1Cc2c(C(=O)NCCNC(c3cccc4ncccc34)=O)cccc2N1 N1(C(C(CC)OCC)=O)CCC(CNC(C2CN(C(C)=O)C2)=O)C(F)(F)CC1 [N-]=[N+]=NCCCC(=O)NCCOCCCNC(c1ocnc1C1CC1)=O c1(C2(C(=O)NCCCN(C(C(CC)SC)=O)C(C)C)CC2)ccc(Cl)nc1 c1(C(=O)NC2(CC=C)CCN(C(=O)C(CC)NC(N)=O)C2)ccc(F)c(F)c1 C(CO)(CC(F)(F)F)NC(C1CC(O)(CNC(c2ccc(C(N)=O)o2)=O)C1)=O c1(C(N(CC(CC)NC(=O)CCF)C)=O)c[nH]c2cc(F)cc(F)c2c1=O c1(C(=O)NCC(CC)(CC)NC(C2CC2C2CC2)=O)cncc(F)c1C N1(C(CCC)=O)CCC2(C1)CN(C(=O)C=Cc1n[nH]c(COC)n1)C2 CCC(O)C(F)(F)C(=O)NCCCN(CCCNC(=O)CC(F)(F)F)C C1(NC(c2ccc(C)nc2)=O)CC(C)CN(C(c2sccc2Cl)=O)C1 n1(CC)nnc2c1CCC(C(=O)NC1CC(F)CN(C(c3csc(C)c3)=O)C1)C2 N1(C(c2c(C)n[nH]c2C)=O)CCN(C(c2n[nH]cc2Cl)=O)CC(O)C1 C1(CNC(c2onc(C)n2)=O)C(C)CCCN1C(=O)C1=CCOC1 CC#CCC(C(=O)NC1CCC2(C(C)C)CC12)NC(=O)C(C)OCCCC C1(NC(C=C(CC)C)=O)CCC1NC(=O)C(=O)NC(C)C N1(C(C2N(C(CNC(CC)=O)=O)CCC(F)C2)=O)CC2CCC(C1)C(=O)N2 CCCC(=O)NC1(CC(=O)NCC(O)CO)CC1 N1(C(C2N(C(CCC)=O)CSC2)=O)C2CCC1C(NC(c1cc(Cl)no1)=O)C2 C1(NC(C2CC(N(C)CC)C2)=O)CCCCCN(C(=O)CN2CC(C)(OC)C2)C1 c1(CNC2C(C(N3CCC(N4CCCCC4)CC3)=O)CCC2)cnc(Cl)cn1 CCCCC(C)C(=O)NC1CCCC1CC(=O)NCCCC1(O)CC1 CP(C)(=O)C(O)C(=O)NCC1=CCN(C(C2(F)CC2)=O)CC1 c1(OC)cc(C(c2nnnn2CC2CC2)NC(C)CS(=O)(=O)CC)cc(F)c1 C1(NC(CCNC(C)=O)=O)CC2(CCN(C(C3CC(C)CC(C)(C)C3)=O)CC2)C1 c1(-c2nnc(COC3CC(CC(=O)OC)C3(C)C)o2)cnn2c1CCC2 c1(OC)ccc(C)cc1CC(N1CCC(C(C)(C)NC(C2C(C)C2(F)F)=O)C1)=O c1(C(=O)NCC2C(NC(C3C(CC)OCC3)=O)COC2)nccc(C)n1 C1(NC(=O)CCCn2ccnn2)CCCC12CCN(C(c1ncncc1Cl)=O)C2 C(=O)(C1=CS(=O)CCC1)NC(C1(O)CCN(C(C(c2ccccc2)OC)=O)C1)C CC1CCN(CC(=O)NC2CCC(OC(C)(C)C)CC2)C1(C)C n1(CC)nc(C(N2CCCC(C(C)C(=O)NCCNC(C)=O)C2)=O)cc1C c1(CC(=O)NCC2(O)CCN(C(C(C)S(N)(=O)=O)=O)C2)c(F)cc(F)cc1F C(c1ccc(F)cc1F)=CC(N1CC(OC)(CNC(c2nc(C)sc2C)=O)C1)=O Cc1cn(CC(=O)N(C2CCN(Cc3cccc4c3OCO4)C2)C)c(=O)nc1O c1(CC(=O)NCC2(F)CC(NC(c3scc(C)c3Cl)=O)C2)cccc(F)c1F c1(C(=O)OCC)cn(C)nc1CNCCC1CCCC1=O C1(C(=O)NC(CC)CNC(=O)CN2C(=O)CN(C)C2=O)Cc2ccc(C)cc2S1 c1(N2CCC(C(F)(F)F)(OC)C2)nc(=NCC2CCCCS2)[nH]c2c1CCC2 N1(C(C23CC(C)(C2)C3)=O)CCC2CN(C(C3CCC(F)(F)C3)=O)CC2CC1 C1(C(=O)NCCCn2cc(CCCCCO)nn2)CC2C=CC1O2 c1(CSCCC(=O)N(CC(C)CNC(=O)CC(C)C2CC2)C)ccccc1Cl c1(CC(c2n(C)nnn2)NCCc2nc(Cl)sc2Cl)cccc(OC(F)F)c1 Cc1nnc2cnc(C(N3CC(CNC(C4CCC(O)C4)=O)CC3(C)C)=O)cn12 c1(C(N(CC(C)(C)NC(C(CSC)OC)=O)C)=O)ccccc1OCC(C)C C12(NC(=O)CCc3ncc[nH]3)CCN(C(c3cnc(C(F)(F)F)s3)=O)CC1C2 N1(C(C2CC(=C)C2)=O)CCC(NC(=O)C(C)Cc2cccnc2)C1(C)C O=S(=O)(c1cc(Cl)cc2cccnc12)NCC1CC(F)C1 C(=O)(N=c1[nH][nH]cc1Br)C1(c2cccc(-c3ccco3)n2)CC1.C(CO)(C(F)(F)F)C(=O)N.C c1(C(=O)NC2C3CN(C(CC(C)N(C)C)=O)C2C3)cn2c(n1)CCC2 N1(C(CCOCCCOC)=O)CCCC(C)C1CNC(c1ocnc1C)=O Cc1nn(C(C)C)cc1C(N1CCC(NC(c2ccccc2C(C)(F)F)=O)C1)=O N1(C(C23N(C(CNC(C=C)=O)=O)CCC2C3)=O)CCCC2(CCCC2)C1 c1(C(N2CCC(Oc3ccccn3)C2)=O)cc2c(nc1O)CCCC2 c1(NC(=O)OC)ccc(S(=O)(=O)NC(C2(c3ccccc3Cl)CCC2)C)cc1Cl C(=O)(C1CCCc2c[nH]nc21)N1CCC2(C(NC(c3c(C)nn[nH]3)=O)C2)C1 C(=O)(C1=C(Cl)CCOC1)NC1C2CN(C(c3ccc(OC)nc3Cl)=O)CC1C2 N1(C(CC(C(C)C)C)=O)CCCC2(CNC(c3ccoc3Br)=O)CCCC12 C#CCC(C)(CC)C(=O)NCC1CCCN(C(=O)CCCS(C)(=O)=O)CC1 c1(C(=O)NC(C(C)NC(=O)CC(=O)N(C)C)C)nc(C(F)(F)F)ccc1F C#CCCCC(C)C(=O)NC1(C2CN(C(c3csc(-c4cnc[nH]4)n3)=O)C2)CC1 C(CC(=O)CC(=O)NCC)N(C(=O)CCC)CC=C.C1CCNC(=O)N1 C=CCCCCCC(=O)NCCCC1(NC(=O)Cn2c(C)cc(C)nc2=O)CC1 CC(O)C(C(=O)N(CC(C)(C)NC(=O)C(c1ccc(F)cc1)CO)C)NC(N)=O c1(CC)nc(C(=O)NC(C)CC2CCN(C(=O)CCCCSC)CC2)c(N)s1 c1(CC(=O)N(C2CCN(C(C(CC)O)=O)C2)C)ccc(NC(C)=O)cc1 Cc1cc(C)n(CCC(=O)Nc2ccoc2)n1.C1C(C)(C)CC2CN1C2 C1(CN(C(C2C(C)CCC2)=O)C)CCCCN1C(=O)C=CCN1CCOCC1 C1(CNC(CNC(CC)=O)=O)CC2COCC2N1C(c1ccc(C(F)F)cc1)=O c1(OC)cnnc(C(=O)NCCOCCCNC(=O)CC2CCC(=O)NC2)c1 N1(C(CSCC)=O)CCC2C(CCN2C(=O)C(C)(C)F)C1 N1(C(COCC(=O)OC)=O)CCC(CCCCCNC(=O)C(O)COC)CC1 Cc1ccc(CC(=O)NCC(C(C)(C)C)NC(C2CCCCO2)=O)c(Cl)c1 C1(C)(NC(CC=CC=C)=O)CCCN(C(=O)CC(C)CCC)C1 C#CC1CCCN(C(=O)C(CCC=C)NC(c2c[nH]c(C)c2)=O)CC1 c1(N2CCC(c3ncn4ccc(C)cc43)CC2)ncccc1S(=O)(=O)N(C)C CS(=O)C=CC(=O)NC1CCCC(NC(C2(CN3CCCC3)CCCC2)=O)C1 C(N=c1nc2c(ncn2C(C)C)c(NCC2COC(=O)N2)[nH]1)c1c(CC)c[nH]n1 C(CC(CC)C(=O)N1CC2(CC(C(=O)NCC3(CO)CC4CC4C3)C2)C1)=CC Cn1cc(C(N2CCC2CNC(=O)C(F)C2CC2)=O)nn1 Cc1n[nH]c(C)c1CNC(=O)C(c1ccoc1)NC(C1CC(C)CCO1)=O N1(C(COCCOCC)=O)CC2CN(C(C3CN4CCC3C4)=O)CCC12 Cc1nc(C(=O)N(C)CC=CC(=O)NCCN2CCCCC2)cs1 c1(NC(COC)CCOC)ncnc(N2CCCC(C(N)=O)C2)c1C c1(C(CC)NC(C)CC2CCOCC2)ccc(F)cc1 C(CC)(C(=O)NCCN(C(=O)C(C)C1CN(C(=O)OC(C)(C)C)C1)C)OCC C1(C(=O)NC(CC)C)CN(C(=O)Cn2cccnc2=O)CC1(F)F N1(C(C(=O)NCCCSC)c2cccs2)CCCC(Cc2ccc(O)cc2)C1 Cc1cc(C(N2CCCC(CN(C(=O)CN3CCC(C)C3)C)C2)=O)c(F)cc1N c1(C(=O)NC2CCN(C(=O)CCc3cncs3)CC2CO)ccc2nc[nH]c2n1 c1(C(CC)NC(C=C)(C)C)cc(OC(F)F)c(OCCC)c(OC)c1 CC(=O)CCCC(C)C(=O)N1CC(C)(C(=O)NCCOCCO)C1 CCC(C)(CCNC(C1CC(C(F)(F)F)C1)=O)NC(=O)CCOC N1(c2nnc(C(CC)(C)C)o2)CC(CNC(c2nc(C)oc2C)=O)OC2(CCC2)C1 c1(C(=O)NC(C2CCN(C(C(COC)C)=O)C2)C)cc(C2CC2)[nH]c1C1CC1 C(=O)(C(C)(C)n1cc(NC(=O)C(c2ccccn2)O)nn1)OC Cc1c(C(N2CC3CC=CC2C3)=O)nc2sccn12 c1(C(=O)NCC(C(C)C)(C)NC(=O)C(C)OCCN(C)C)ccc(F)cc1O c1(CNC(C2N(C(c3cnc(OC)nc3)=O)CCC2)=O)c(C)nn(C)c1C Cc1nc(NC2(CNC(C3CCCC(C)C3)=O)COC2)[nH]c(=N)n1 Cc1cnoc1C(=O)NCC(C1CCCN1C(=O)Cc1ccccn1)(C)C C(CC(C)C)(C(=O)N(C)CC1(O)CN(C(c2cncc(C)n2)=O)C1)OC N1(C(C2C(OC)C2)=O)C2CCC1CN(C(C1OCCC1(C)C)=O)C2 c1(C(N2C(C(N(C(c3ccccc3)C)C)=O)CCC2)=O)cnc(C(C)(F)F)cn1 C1(C(=O)OC)CCN1C(=O)CNC(=O)CNC(=O)Cn1nccn1 N1(C(C2(CC)CC2)=O)CCC2(CC1)OCCCC2NC(C1COCC(C)(C)O1)=O C1(CNC(C2(OC)CCSC2)=O)C(C)CCCN1C(=O)CN1CCCCCC1=O C#Cc1ccnc(C(=O)NCC2CCC(C)CN2C(c2ccc(C(C)C)o2)=O)c1 c1(C(=O)NC(c2ccccc2OC)CNC(C2C=CCS2)=O)cc(F)cnc1O C1(CNC(=O)CCn2ccnn2)CC2CCC(C1)N2C(c1cc2sccc2[nH]1)=O C1(F)(CNC(c2c(CC)noc2)=O)CC2CCC(C1)N2C(=O)C(CC)C(F)(F)F c1(C(N2CCN(C(c3n(CC)ncn3)=O)C(CO)C2)=O)ccc2c(c1)N(C)CC2 C(C)(CCC(C)(C)C)N(CC(=O)NS(c1c(OC)ccs1)(=O)=O)C(C)C CCC(CNC(=O)C(N1CCCC1)C1CC1)N(C(=O)CCOCC1CC1)C C1(C(=O)NC2CC2C2CC2)CC2CCC(C1)N2C(c1cc2ccccc2[nH]1)=O C1(C(C)C)C(C(=O)NCc2ccnn2C)CCN1C(=O)CN1CCNC1=O c1(C(=O)NC2C(NC(C(c3cccnc3)OC)=O)CC2)cc(=O)n(C)cn1 C=CCCC(C(=O)NCc1nc(CC)no1)NC(C1C=CCCCC1)=O C1(C)(NC(C2C(OCCC)CCCC2)=O)CCN(CCCC2CCOCC2)CC1 N1(C(C2(C)CCCCO2)=O)CCC(O)(CCNC(=O)CCc2ccc(Cl)s2)CC1 n1(C(C)C)nc(C2CCOC2)nc1C1CC(=O)N(C)C1 N1(C(CNC(=O)OC)=O)CCC(CCCCCNc2sc(C)cc2Cl)CC1 Cc1ccc(F)c(Nc2nc(C(=O)N(CC3=NOC(C)C3)C)nc(=N)[nH]2)c1 C(C(C)(C)C(=O)NCC1CC(NC(C2(O)CCCC2)=O)C1)N(C)C N1(C(=O)CCOc2ccccc2)CC2CN(Cc3cc(Br)ccc3Cl)CC2C1 c1(SC)cnn(C)c1C(=O)NC(C)CN1CCN(C(C2(C)CCOCC2)=O)CC1 O(NC(=O)CC(C(F)F)NC(=O)C(C)SC(C)C)CCCCC c1(CC(N2CC3(CCN3C(=O)CCC3OCCO3)C2)=O)ccc(F)c(Cl)c1 c1(C(=O)NCC(C)(C)CNC(=O)Cc2cc[nH]n2)ccc2n[nH]cc2n1 Cc1occc1CNC(=O)C(C)(C)NC(C1CCSCC1)=O CCCC(C)CC(=O)N1CC(O)(C(C)NC(=O)CN(C)Cc2ccc(C)cc2)C1 c1(C(=O)NCCNC(C2N(S(CC)(=O)=O)CCC2)=O)cccc2ccoc12 N1(C(c2cc(F)ccc2F)=O)CCOC2CN(Cc3csc4cncn34)CC12 C1(CCC(=O)NCCc2cccs2)CCCCN(C(c2n[nH]cc2Br)=O)C1 C1(F)(C(N(C(C(N2C(C(=O)NC)C=CC2)=O)C)C)=O)CC=CCC1 C1(C(CNC(c2ccsc2)=O)(C)C)CCCCN1N(CC(=O)NCCCC)C.C(C)=O Cc1ccnc2c(C(=O)NC3CCC3CNC(C3CC(=O)NC(=O)N3)=O)cnn12 N=c1[nH]cncc1C(=O)NCc1ccsc1C(=O)NC1CC(CC2CC2)C1 CC1CCN(C(C2(C3CC3)CCC2)=O)CC1NC(=O)Cn1cc(C(F)(F)F)cn1 N1(C(CC2OCCN(C(C)=O)C2)=O)C(C)CN(C(c2sccc2F)=O)CC1C Cc1ccc2[nH]cc(CC(=O)N(C3CN(C(C4CCC(C)NC4=O)=O)C3)C)c2c1 N1(C(C2(C#N)CC=CC2)=O)CCCCC(CCC(=O)NC2(CO)CC(F)(F)C2)C1 N1(C(c2c(=N)[nH]cnc2)=O)CCC2C(CCCN2C(=O)Cc2ccc(O)nc2)C1 C1(C)(CNC(C2C(CNC(c3cn(CCC)nn3)=O)CC2)=O)CSC(C)=N1 CC1CC(C(=O)NCCOC2CCN(C(=O)CN3CCN(C)CC3)CC2)CCO1 c1(C(N2CCCCC(CNC(c3cc(C)[nH]n3)=O)C2)=O)cc2ccoc2cc1F N(C1CCc2ccccc21)(C(=O)Cn1c(O)nc2ccccc12)CCC C1(CNC(=O)CCOC2CC2)CN2CCCCC2CN1C(=O)CCc1cncs1 C1(C)(C(=O)NCCNC(c2c(C)nc[nH]2)=O)CCC(O)CC1 N(C(=NCCSC)NCCN1CCC(C)CC1)CCN(CC)CC c1(CC(=O)NC2CN(C(CC=CCC)=O)C2)cc(C(C)C)no1 CCCCCC(C)CC(=O)N1CC(CCCCNC(C23CCOC2CCOC3)=O)C1 CC(C)C(O)C(O)C(=O)Nc1ccc2[nH]ncc2c1 N1(Cc2nc(CC)on2)CCC2C(CCCN2C(c2cc(C)n(C(C)C)n2)=O)C1 N1(C(c2cc(SC)ncc2)=O)CC(NC(=O)C(c2ccccc2)F)C(N=[N+]=[N-])C1 N1(CCC)C(=S)NC(c2cnc(C(C)C)o2)C2=C1C(C)N(C)C2=O c1(C(CNC(=O)C(c2ccc(Br)cc2)=O)=O)cc(Cl)cc(Cl)c1 c1(C(=O)NC2C(C)(C)C2)ccc(CNC(C2CN(C(=O)N(C)C)C2)=O)nc1 N1(C(CC2=CCN(C)CC2)=O)CCC2(CCCN(C(=O)C=Cc3cc[nH]c3)C2)C1 N1(C(COCC(=O)OC)=O)CCN(C(c2coc3c2CSC3)=O)CC(O)C1 C1(OC)CN2CCCC2(C(=O)NCC2CN(C(=O)COC(F)(F)F)CCN2C)C1 c1(C(N2CCN(C(C=CSC)=O)CC2CF)=O)cccc2[nH]ncc12 C1(C(N(CCCC(=O)NCCc2cnc(C)o2)CCCO)=O)CCC2(CC2)C1 N1(C(CC(C)(C)OC)=O)CC2(CCCC2NC(=O)CNC(c2ccsc2)=O)C1 c1(-c2nc(COC)sc2)ccc(F)c(C)c1C(=O)Nc1cc(N(C)C)no1 c1(CN(CC(=O)NC(CCCNC(c2c(C)nc[nH]2)=O)C)C)cccc(Cl)c1 C(=O)(C(CO)c1ccccc1)NC(C1CN(CC=CCl)C1)C C(=O)(N1CC(O)CCO1)C1N(C(c2cncc(OC)n2)=O)CCCCC1 c1(C(=O)OC)cc(Br)c2[nH]c(=NC(C)C(C)C)[nH]c(=N)c2c1 N1(C(C(c2cnc(C)s2)NC)=O)CCCC(F)(F)C1 C1(C(=O)NC(C2CC2)=O)CCCO1.O=C1CN(C(=O)COCCCF)CCN1 C1(C)(C(=O)NC2(CC=CC(N3CC(C(=O)OCC)C3)=O)CCC2)CCCCC1C c1(C(N2CCC(C)C2C(=O)N(C)CC2CN(C)C2)=O)c[nH]c2cnccc12 N1(C(C(CCNC(CC(CC)C2CC2)=O)OC)=O)CCn2ccnc2C1C c1(C(=O)NCC(=O)NC2CC2)occc1CC(C1CC1Cl)=O N1(C(C(C2CC2)OC)=O)CC=CC1C(=O)NCCCOCC1CC1 O=C(C1=NOCC1)NC1CCOCC1NC(c1ccccc1N1CCCC1=O)=O c1(C(N2CC(C(N(CC)Cc3ccccc3F)=O)OCC2)=O)cc(C)n(C)c1C N1(C(C=CC(C)NC(c2c[nH]cc2C2CC2)=O)=O)CCC2OCCC2C1 C1(CCOC)CN(C(c2ccnnc2O)=O)CCN1C(=O)CC1C=CS(=O)(=O)C1 c1(NCc2n(C)ncc2S(C)(=O)=O)nccc2ccncc12 C1(CCCNC(C2CC2C(F)(F)F)=O)CCN(C(C2(C3CC3)CCCO2)=O)CC1 C1(NC(c2ccc(CC)c(Cl)c2)=O)CC2CC1CN(C(=O)C(COC)OC)C2 c1(-c2cccc(CC(=O)OC)c2)ccc2c(c1NCC1(C(F)(F)F)CC1)OCO2 C1(C(N(C(CNC(c2cccc(C(C)C)n2)=O)C)C)=O)C2CC3C(C2=O)C13 C(=O)(CC(=O)N(C)CC1(O)CN(C(c2cc(-c3ccncc3)no2)=O)C1)OC Cc1cnc(NC2CCCC(C(C)(C)C)CC2)c(S(=O)(=O)NCC2(F)CCC2)c1 C1(NC(C(N2CCC(O)CC2)C)=O)CCC(O)CN(C(=O)CCC(F)(F)F)C1 C(=O)(C(=O)CC(C)C)NC(C(=O)N(C)Cc1c(C)occ1)C1CC1 C1(NC(=O)OCC=C)CCN(C(=O)C(=O)N(C)C)C1.C1(C)C(=O)N1C1CC1 CCC(CC(=O)NC1CC2CN(c3c(F)cccc3[N+](=O)[O-])CC12)CC(F)(F)F C(CCCC(F)(F)F)NC(C(CN(C)C)NC(c1n[nH]c(CC)c1C)=O)=O C1(NC(c2ccc(SC(F)(F)F)o2)=O)COCC1NC(C1CCOC1)=O C(C)(C)(CC(N)=O)NC(CC1(N(C(C(C)N(CC)CC)=O)C)CC1)=O C(=O)(C1CCCc2c(Br)cccc21)N1CCN(CCCC)CC1 n1(CC(C)C)ncc(C(=O)NCC(CNC(=O)CN(C(=O)C(C)C)C)CO)c1C CC1CC(NC(c2conc2C2CCC2)=O)CN1C(=O)CN(c1ncccn1)C c1(C(C(=O)NC2(C)CC2)N(CCCO)CC2CCOC2)ccnc(Br)c1 c1(C(N2CC(NC(C#CC3(C)CC3)=O)CC3(C2)CC3)=O)ccc2c(c1O)CCC2 C1(C(N2CCC(N(C(=O)C(C)=CC3CC3)CCC)C2)=O)CC12CCCC2 c1(COC)nnc2n1CCN(Cc1cccc3nn(C)nc13)C2 N1(C(=O)NC(c2cn3c(n2)CCCC3)C)COC2CCCCC2C1 CCCCCCCCCC(CC)C(=O)NC1CC(CC(=O)NCC(F)(F)F)C1 N1(CCSC)C(=O)NC(c2cc(S(N)(=O)=O)cs2)C2=C1CC(C)CNC2=O CCC(N=c1cc(NCCc2cc(C)on2)nc(C(C)C)[nH]1)C1CC1 N1(C(c2cc(C3(C)CC3)n[nH]2)=O)CC(NC(c2n[nH]cc2[N+](=O)[O-])=O)CC1(C)C Cn1nc(Br)c2c(N3CCCC(N4CCCNC4=O)C3)ncnc12 c1(C2(C(=O)NC(C(C)C)CN(C)C(=O)C3CC3)CC2)cccnc1Cl N1(C(C(C)(C)CC2CC2)=O)CCC2CCCN(C(=O)Cn3nnc(=O)[nH]3)C2C1 Cc1[nH]ccc(=NC(=O)Nc2cc(C(=O)O)c3cccnn23)c1Cl C1(NC(C(CCC2CC2)NC(C2CCC(C)(C)CC2)=O)=O)CC(C)(C)OC1(C)C CCC(=O)CCC(=O)N(C1(C(=O)N(C)CC2(C#N)CC2)CC1)C c1(C(=O)NCC2COCCN(C(c3c(C)c[nH]c3)=O)C2)ccc2c(c1)COCC2 c1(C(=O)OC)ccc(CCNC2CC(OC)C2)cc1 CC1=C(C(=O)NCCCCNC(C2(C#N)CC2C(F)(F)F)=O)CCC(C)(C)C1 c1(CNC(c2cccc(I)c2F)=O)ccc(F)cc1O.c12ncc(cn1)CCN2 C1(C(N2CCC(C)C(NC(c3c[nH]cc3Br)=O)C2)=O)(CC)CCC(F)(F)CC1 c1(C(=O)NCC(CC)N(C(=O)C(C)N(CCCCO)C)C)ccc(=N)[nH]n1 c1(OC)ccc(Cl)c(Cl)c1C(N1CC2(NC(=O)CC3CCOC3)CCC1CC2)=O c1(N(C2CN(C(=O)OC(C)(C)C)C2)C)c(C#N)cnn1-c1cccc(Br)c1 C1(NC(C(CC)C)=O)CCN(C(C2CC3(CC(OCC)C3)C2)=O)C1(C)C C1(NC(C=Cc2ccc(OC(C)C)cc2)=O)CCc2nncn2C1 c1(-c2ccc(C(N3CC(C(F)(F)F)(OCC)C3)=O)o2)ccc(C(C)C)cc1 CC(C)CC(C)(CNC(c1cccc(O)n1)=O)NC(=O)C(C)c1ccsc1 Cc1ccc(CCCNC(c2ccc(C)c(F)n2)=O)cc1C CCC(C(=O)N(C1CC(NC(=O)Cn2cnnn2)C1)C)c1ccccc1 C1(NC(=O)C=Cc2ccncc2)CC2(CCCCN2C(C2CCCCC2)=O)C1 C12(NC(CCCNC(C)=O)=O)CCN(C(c3cc(C4CC4)ncn3)=O)CCC1C2 CCCCC(CC)CC(=O)N1CC(NC(c2cnn3c2CCCC3)=O)CCC1C c1(C(C(N)=O)NC(=O)NC(c2ccc(NC(N)=O)cc2)C)ccc(Br)cc1 c1(NCCC(=O)NC(C)CN(C(=O)CCc2cccnc2)C)ccccc1 C(CNC(=O)CCc1cc(Cl)cs1)(CC(F)(F)F)NC(C(C)c1ccco1)=O C(=O)(CCC(C)SC)N(CC)Cc1ccccc1.C1(=O)CC(N)CN1 c1(OCC(N2CC(CNC(CC=CCC)=O)C2)=O)ccccc1C(F)(F)F c1(CNC(CCSCC)=O)nc(CNC(c2ccsc2OC)=O)cc(O)n1 CCC(CCCC(=O)NC(C)CCCCO)NC(c1n[nH]c2ccccc12)=O Cc1c(OCc2nc(C3CCOC3)n[nH]2)cccc1[N+](=O)[O-] N1(C(CCCSC)=O)CC2C(CNC(c3ccc(N(C)C)cc3)=O)C2C1 CC(=O)C(C)CC(C)C(=O)N1CC(NC(C23CCC(C2)C3)=O)C2(CCCC2)C1 C1(ONC(CN(C(=O)CCCNC(C)=O)CC)=O)CCC(O)CC1 C12(C(N(C3CCC(=O)NC3)CC)=O)CC(CN(C(C3C=C(C)CS3)=O)C1)C2 c1(C(=O)NC2CCCCN(C(c3cc(Cl)cnc3O)=O)C2)c(F)ccc(F)c1F c1(OC)cnc(F)cc1C(N1CC(CNC(c2cc3sccc3s2)=O)C(O)C1)=O c1(C(N2CCC(CN(C(C(CC)C(C)O)=O)CC)CC2)=O)c(C)cc(C)oc1=O CN1CCC(C2CCN(C(C3CCOC(C)(C)C3)C(=O)NC(C)(C)C)C2)CC1 CC(C)C(C(=O)N1CC(CNC(=O)Cn2cnnc2)C1)S(=O)(=O)C1CCCCC1 C(C)(CC(C)NC(=O)C(=O)NCC(F)(F)F)NC(C(C)=C(C)C)=O C1(NC(C(C)=O)=O)CCCC2CN(C(c3cc4cccc(C)c4[nH]3)=O)CC12 c1(N(CC(=C)Br)C)nc(NCC2CCN(CCOC)CC2)c2ccsc2n1 N1(C(CN(CC)CC2CCSC2)=O)CCC(C)(C(=O)NC2CC2C(C)C)CC1 Cc1ccc(CN(C2CCCN(C(=O)CCC(C)C)C2)C)nc1 c1(C(=O)OCC)n[nH]c(=NC2CN(C(=O)CCOC3CC3)CC2(C)C)s1 C1(C(=O)NC2CCCC(CNC(c3nc(C)[nH]n3)=O)C2)CC(=O)NC(=O)C1 C1(NC(c2ccc(=O)oc2)=O)CCN(C(=O)C(F)(F)C2CC2)CC1O c1(OC)ccc(S(=O)(=O)NC2C3CN(C(c4ccc[n+]([O-])c4)=O)CC23)cc1 C#CC(C)(C)C(=O)NCc1ocnc1C(=O)NC1CCCC(C(=O)OC)C1 c1(CN(C(C(=O)NCCC(=O)OCC)c2cncs2)C)cccc(F)c1F c1(OC)cc(CN(C=O)C(C)Cc2ccc(F)cc2F)c(OC)cc1Cl n1(CC)nc(C)c(C(=O)NC2CCN(C(=O)COC3CCCC3)CC2)c1Cl c1(C(N2CC(C)(NC(C3CCOC3C(F)(F)F)=O)C2)=O)n[nH]c2cc(Cl)ccc12 N1(C(c2c(CCC)[nH]cc2)=O)CC(NC(c2cc(Cl)ns2)=O)C(CC)C1 Cc1cc(Br)ccc1COC(c1cccnc1C(C)C)=O c1(C(CN(CC(C)(CO)c2ccccc2)CCO)O)ccc(C(F)(F)F)cc1 N1(C(CNC(CCC)=O)=O)CC=CC1(C)C(=O)NCC(O)CC c1(COC)nc2ccccc2[nH]1.C(CC(=O)N(C)CCNC(=O)CSC)OCC N1(C(c2cnc(OCC)s2)=O)CC2CCCC(C1)N2C(=O)C(C)CC(C)C N1(C(CSCCC)=O)CCC2(CCCC2NC(c2cc(C)ns2)=O)C1 N1(C(C2CCC(CC)CC2)=O)CC2CCC(C1)C2NC(=O)C=Cc1cccnc1 O=C(CCC(F)(F)F)N1CCCC(F)(C(N2CC3CCC3(CO)C2)=O)C1 C1(NC(C(C)Sc2cccc(C)c2)=O)Cc2ccc(C)cc2C1 c1(CC(N2C(C(C)NC(C(CC)COC)=O)CCC2)=O)cc(Br)ccc1C CC(C)S(=O)(=O)C(C)C(=O)N1CCCC(CO)(CNC(c2cc(O)nn2C)=O)C1 C12(NC(CC=C=C)=O)CC3CCC(C1C2)N3C(=O)C(n1cc2ccccc2n1)C CC1CCCCN1CCCCC(N1C(CC(=O)NC(=O)CO)CC1)=O C=CC(F)(F)C(=O)N(C1CC(C(=O)NCC2CC(O)CN2C)C1)C N1(C(C2(C=C)CCC2)=O)CCN(C(=O)C(N2C(=O)CCC2=O)C)CC1 c1(OC)ccc(C2(C(=O)NCC(C)N(C(=O)C(F)n3cccn3)C)CC2)cn1 C1(C(=O)NC2CC(O)(CNC(C3C(CC)C3)=O)C2)CNC(=O)CC1(C)C N1(C(CC(C(C)OC)NC(c2ccc(C(C)=O)o2)=O)=O)Cc2c[nH]nc2C(C)C1 c1(C(=O)NCC2(COC)CN(C(C3CC3C3CCCC3)=O)C2)ccc([N+](=O)[O-])o1 C1(C(=O)NCC(C(C)C)NC(C(CC)Sc2ccccc2)=O)CCC(=O)N(C)C1 N1(C(c2ccc(SCC)nc2)=O)CCC2CN(C(=O)C=Cc3cc[nH]n3)CC12 C(C)(CC(=O)NCCOCCOC)N(C(CSCC#C)=O)C c1(C(=O)NCC2(OCC)CN(C(COCCC=C)=O)C2)ncc(C)cc1F Cc1oc([N+](=O)[O-])cc1C(N1CCC(C)C(NC(=O)CCS(N)(=O)=O)C1C)=O N1(C(CCC=C)=O)CCCC(C)(CNC(=O)C(C(C)O)NC(=O)NC2CC2)C1 C(C1CCCC1)=C(C)C(=O)NC(C1(CNC(=O)C(C)OCCN(C)C)CC1)C c1(C(N2C(CN(C(=O)CC3CC4CC4C3)C)CCC2)=O)ncc(C#N)cc1Cl C1(N=[N+]=[N-])(C(=O)NC2C(C)CCCCC2)CCN(C(=O)Cn2cc(CO)nn2)C1 C1(C(N(C)CC2(O)CN(C(c3c(Cl)cn(CC)n3)=O)C2)=O)CCn2nnnc2C1 CC(C)C(C(C)NC(c1conc1C(F)(F)F)=O)NC(=O)C=CCF c1(Oc2n(C)ccn2)cccnc1CNC(C1COC(C)(C)C1)=O C(=O)(CCCC(C)=O)N1CC(OC)C(NC(c2nn(C)c(Cl)c2Cl)=O)C1 C(=O)(C(C(C)(C)C)NC(c1cnncc1C)=O)NCC(COCC)C C(=O)(C1=Cc2ccccc2OC1)NCC(C)NC(=O)C(C)C(C)c1ccc(F)cc1 C(CCN(C)C)(C(=O)N(C)Cc1ncc(C)o1)NC(C1ON=C(C)C1)=O c1(CCNC(=O)C(N2CCCC23CCC3)C2CC23CCOC3)cc(Cl)cc(Cl)c1 C(CCCCC(=O)NCC1CC1C)N(C(Cc1cn(CC)nn1)=O)C Cc1nc(C2CC2)sc1C(=O)NC12CC1CN(C(C1CC1F)=O)C2 N1(C(C2CCC(NC(C(C)(C)n3cncn3)=O)C2)=O)CC2CCC2(C)C1 CC1(C)CN(C(C2COCCN2C=O)=O)CC(CNC(=O)C2=COCCC2)O1 c1(C(=O)NCCC2CCCN(C(CCc3cnn(C)n3)=O)C2)cccc(Cl)c1N C1(CC(=O)NCc2c(C)ncs2)CN(C(=O)CCc2cnn(C)c2)CC1C c1(CC)cscc1C(=O)N(CC(C)C)CCNC(C)(C)C N1(C(C2(C)CC2(F)F)=O)CC(N=c2nc(C3CCCC3)[nH]s2)C1 C(C#Cc1cccc(Cl)c1)N(C1CCCN(C(CCCc2ccc(C)s2)=O)C1)C c1(-n2cc(CCN(C)C(c3nsnc3O)=O)nn2)cccc(CO)c1 Cc1cc(C)c(C(=O)CCCC(=O)NC(C(=O)O)C2CNC2)c(C)c1 c1(C(=O)OCc2cc(C(=O)OC)c(OC)cc2)cc(N)c(F)c(F)c1Cl C1(CC(=O)N(CC(C)NC(C2(CSC)CCC2)=O)C)SC(=N)NC1=O c1(C(=O)NCC(CNC(=O)Cn2cnnc2O)OC)cccc(N)c1O N1(C(c2c(C)cns2)=O)CCCN(C(C2CCN2S(C)(=O)=O)=O)CC1CO CC(C)CC(C)CC(=O)NC1(C)CCCN(C(c2ccc(F)c(C(F)F)c2)=O)C1 N1(C(COCCCC(C)C)=O)CC2CCCN(C(C3CC4COCC4C3)=O)C2C1 C12(C(=O)NCc3ccn(CCC)n3)CCCCC(F)(C1)C2 C1(C(=O)NC(c2ccc(C)nc2)C)C2CC3C(C2NC(c2cnc(O)o2)=O)C13 c1(CCCC(N2CCC(N(C(C(C)N(C(C)=O)C)=O)C)C2)=O)ccc(C)c(C)c1 CN1CCN(C(C2CC2F)=O)C(CNC(C2CC3CCC2C3)=O)C1 c1(OCCNC(=O)CN2CCN(Cc3cccnc3Cl)CC2)cnc(Cl)c(Cl)c1 c1(CC(N2CC(C)C(NC(c3cccc(=O)n3C)=O)C2)=O)cc(F)cc(F)c1 C12(NC(CC3C(=O)NC(=N)S3)=O)CCCC1CN(C(c1cncnc1)=O)C2 c1(NC(C)=O)ccc(C(=O)NC2CN(C(=O)CSc3ccccn3)CC2O)cc1 CCCCCC(O)CC(=O)N(CCCNC(C1CCN(C)C(=O)C1)=O)CC C1(C(N(CCC(=O)NC)CC)=O)CCN(C(=O)C(C#N)C(C)(C)C)C12CCC2 Cc1noc(C)c1CN1CCC(NC(c2cc(Br)c[nH]2)=O)C1 CC1CCCN(CC(C)NC(c2ccc(N3C(=O)CCC3C)cc2)=O)C1 C(=O)(C1=CCCCO1)NCCCC(C)(C)NC(c1cc2c(s1)CCC2)=O CS(=O)(=O)c1ccc(OCCOC(C2CC2Cl)=O)c(C(=O)O)c1 c1(C(N2CC(NC(CC(CC)(C)C)=O)C(C)CC2)=O)sc2ncccc2c1N C1(C(=O)Nc2cc3c(nn2)CCCC3)CS(=O)(=O)C12CCCC2 Cc1cc(C(=O)N(CC(O)CNC(=O)CC2CNC(=O)C2)C)nc(O)n1 CCCCC(CC)CC(CNC(c1c(C)nn(-c2ccccc2C)c1C)C)CC C(=O)(CCCC(CC)NC(=O)CCc1cc(C)on1)N(CCCC=C)C c1(C(=O)NC2CC(CNC(C(CC(=C)C)OC)=O)C2)cccc2nncn12 C(=O)(C(C(C)C)Nc1ccccc1)NC(CC)CNC(C1C(C(=O)OC)C1(C)C)=O c1(C(=O)NC2CCC(F)(CNC(CC(=C)C)=O)C2)cc(F)cc2ccccc12 c12ccc(cc1)C1(CC1)C(=O)NC2.c1(NC(CC=C)=O)ccnn1COC c1(C(N2CC(CNC(C3CC(=C)C3)=O)C(C)CC2)=O)ccc2c(c1)CCCCN2 N1(C(COc2cc(C)on2)=O)CC(NC(=O)C=CCF)CC1(C)C c1(C(=O)NC2CCCC(CNC(CCC(CC)C)=O)C2)cc(S(N)(=O)=O)cs1 c1(C(N2CC(NC(C=Cc3cc(C)no3)=O)C(O)C2)=O)c([N+](=O)[O-])c(C)nn1C C1(C(=O)NCCCC=C)(CC)CCN(C(c2cccc(OC)c2O)=O)CC1 C1(C(N2CCC(NC(c3c(CC)n(CC)nn3)=O)CC2)=O)OCC2CCCC12 c1(C(N2CCCC(NC(C=C(C)C(=O)O)=O)C2)=O)cc(C)c(F)cc1Br c1(CN2CC(C(=O)Nc3cccc(-n4cncn4)c3)OCC2)c(Br)cncc1Br c1(C(CNC(c2c(CC)n(C)nc2)=O)=O)ccc(Cl)c(Cl)c1 Cc1ccc(Cl)c(C(=O)NC2COCC2NC(C2COCCO2)=O)c1 c1(CC(N2CC3C(N(C(=O)C(O)CC4CC4)C)C3C2)=O)cc(F)c(F)cc1F CC(CCC(C)(C)C)C(=O)N(C)CC1CCCN1C(c1csnn1)=O N1(CC)CCN(C(=NCc2nncn2C)NCC(C)Oc2ccccc2)CC1=O C(CC(=O)NC12CC(C)(C1)C2)(C(C)OC)NC(c1cncc(OC)c1)=O c1(OC)ccc(Cl)cc1NC(N1CCC(C2CCCN2C)CC1)=O c1(OC)cc(C(N2CCN(CCNC(=O)C(F)=C3CCCC3)CC2)=O)ccc1O N1(C(C(C)=CC)=O)CC(C)(CNC(=O)CCCOc2ccc(F)cc2)CC1(C)C C1(CNC(C2(CC(C)C)CCC2)=O)CC2CC1CN2C(C1CCOC1)=O CCC(C(=O)NC1CC(F)CN(C(=O)C(=O)NCC(F)F)C1)C(C)(C)CC c1(CNC(=O)NCc2c(C)cc(Cl)cn2)nccc2cc(Br)ccc12 CCC(C(=O)NCCn1cc(C(N2CC(CC)(CO)C2)=O)nn1)C(C)C n1(CC)cc(CCNC(=O)C(CC2CCCC2)NC(=O)CN=[N+]=[N-])cn1 Cc1ccc(-n2nccn2)c(C(=O)NCCn2cc(-c3ccncc3)nn2)c1 N1(C(C2C(C)(C)C2)=O)CCCC(n2cc(CCNS(C)(=O)=O)nn2)CC1 C1(CNC(C2CCC(NC(c3c(C)nc[nH]3)=O)C2)=O)CCC(=O)NC1 c1(C(=O)NCC2(C)C(NC(c3n(CC)ncn3)=O)CCC2)cc(Cl)cc(Cl)c1 C(CC(=O)NCC(C1CCC1)NC(C1CC1(F)Cl)=O)NC(C)=O c1(C(=O)NC2(C)CN(C(CN(C3CCC3)C)=O)C2)nccc2cc[nH]c12 C=C1CCN(C(=O)CCOCCC)C(C(=O)NC2CCCCC2OC)C1 C1(C(N(CCC#C)C)=O)CCN(C(c2cncc(C#N)c2)=O)CCO1 c1(N2CCN(C)C(CNC(c3ccnn3C)=O)C2)ncc([N+](=O)[O-])c(=N)[nH]1 c1(C(N2CCC(C(N(C)Cc3cccc(Cl)n3)=O)CC2)=O)c(O)cccc1O C1(NC(c2ccc(C(F)(F)F)cn2)=O)CC12CC(NC(C1(F)CC1)=O)C2 CC(C(=O)N1CC(N2CCCC2=O)C1)(C1CCC1)NC(C1(c2cc[nH]n2)CC1)=O N1(C(CC(C=C)C)=O)CC2COCC(C1)C2NC(c1cccc(C2(C)CC2)c1)=O c1(C(N2CC(NC(CCOCC#C)=O)C(C)CC2)=O)cc2cccnn2c1 CC(C)CC(F)C(=O)NC1CC(C)(NC(=O)C(C(C)C)c2ccn(C)n2)C1 c1(C(=O)NCCC(C)N(C(=O)C(C2CCC2)C2CCC2)C)cccn2nccc12 c1(C(=O)OCC)ccc(N2CC(CNC(=O)CCCCCSC)C2)nc1C C#CCCCCCCN=c1cc(C(=O)OC)[nH]cc1Cl C1(C(=O)NCC(C#C)CC)CC2CC1CC2NC(C12CCC(OC)C1C2)=O c1(C(=O)NC(CNC(CCSC)=O)C)cnn(C)c1S(C)(=O)=O CCC(C)CC(C(=O)NCC1(C2CC2)CCCO1)NC(=O)CN(C)C C(=O)(C1=CCCC1C)N1CCC(C(CO)NC(c2c(C)ccnn2)=O)CC1 Cn1cc(C(N2CCCC(NC(=O)CCC3CCOC3)C2)=O)c(=O)n(C)c1=O c1(C(=O)NCC(CNC(C2(C)CCCO2)=O)OC)c(C)ccc(C)c1N C1(C#N)(C(=O)NCC2(NC(c3nc(C(C)C)oc3)=O)CCC2)CC12CCOCC2 c1(C(N2CCC(CN(C(c3c(C)oc(Br)c3)=O)C)C2)=O)ncnc(O)c1F N1(C(=O)CCc2cccc(O)n2)CC2CCN(C(=O)CCc3cn[nH]c3)C2C1 C1(NC(C(COC)NC(=O)C(C2CC2)SC)=O)CCC(C2CC2)C1 C1(CS(=O)(=O)NC(C23CC(CO2)C3)C)CC2(CO1)CC(F)(F)C2 CC1(C)C(CNC(=O)CC2CCCC2(F)F)CCN1C(C1CCCNS1(=O)=O)=O CC1CCN(C(=O)C(=O)NC2(C)CCN(C(=O)Cc3nc(Cl)cs3)C2)CC1 C1(CNC(=O)CN2CC(NC(N3CCCC3)=O)C(O)C2)CCc2nccn2C1 C1(NC(c2c(OC)noc2C)=O)CC2CC(NC(C3CCC(F)(F)C3O)=O)C1C2 CC1CN(C(C2(C(C)(C)C)CCC2)=O)CCC1CNC(c1ccc(F)s1)=O C(CCC(=O)N(C)CC1CCC(C)C1)NC(=O)OC c1(C(N2C(CO)CC(NC(c3ccon3)=O)C2)=O)ccnc2ccccc12 C(=O)(NNc1ccc2ccccc2c1)c1ccc(S(=O)(=O)NC)cc1 C(CC(=O)NCC(CC1CC1)CO)(C1CC1)NC(C=CC=CCC)=O Cc1[nH]cc([N+](=O)[O-])c(=O)c1C(=O)NC1CCC1NC(=O)C(C)c1ccsc1 c1(C(N2C(CNC(C(C=CC)O)=O)CCC2)=O)nc2ccccn2c1F C1(C(=O)NC(C)Cc2ccnn2C)CCC2(CC2)N1C(c1cccnc1)=O c1(C(C(C)C)NC(=O)CC2COCC(C)(C)O2)nc2ccccc2[nH]1 CCC(C)(CCNC(=O)C=CSC)NC(=O)Cc1cc(C)nn1C N1(N(CC=O)CCOC)CC=CC(O)C1.C1(C=O)CCSC1 c1(Cn2cc(CSCC)nn2)ccc(C(N2CC(C(F)(F)F)(OC)C2)=O)cc1 N1(C(=O)NC2CN(C(=O)OC(C)(C)C)C3C2C3)CC2CC1CN2C1CCC1 C1(CC)(CNC(C2CCCC(CC)CC2)=O)CCCC(=O)N1 C1(C(=O)NC2(C#C)CC(=O)C2)CCCCN(C(c2cccc(C)c2C)=O)C1 c1(C(N2CCC(O)(CN(C(=O)C=CBr)C)C2)=O)csc2c1CCCC2 N1(C(C(CC)(C#N)CC)=O)CC(NC(=O)C(F)OC(F)(F)F)CC12CCCC2 N1(C(C2=C(C)CCC2)=O)Cc2[nH]nc(C(=O)NCC3OC(=O)CC3(C)C)c2C1 [N-]=[N+]=NC1CN(C(C2CN3CCN2CC3)=O)CC1NC(C1(N2CCCC2)CC1)=O c1(CC(CO)NCc2cc(COC)on2)ccccc1F N1(C(C=C(C)C)=O)CC2CCC(NC(=O)CCCc3cccs3)CC2C1 C(=O)(CCCCCF)NCC1C(NC(C2CC(C)OC2)=O)CCC1 c1(CC)cncc(C(N2CCCC2(C)CNC(=O)Cc2sc(C)cc2C)=O)c1 C1(C(=O)NC(C2CCN(C(c3cc(O)ncn3)=O)CC2)C)CCn2nnnc2C1 CS(=O)(=O)c1ccnc(NC2CN(C(=O)C=CI)CCC2C(F)(F)F)n1 CC1CN(C(=O)C(F)(F)c2cscn2)CCC1NC(=O)Cc1csc(NC=O)n1 n1(CC(=O)NC(C)CCN(C)C(C23CC(F)(C2)C3)=O)cnc2sccc2c1=O CN1C2CCC1CN(C(=O)CC=CCNC(=O)C1=CCCSC1)C2 CC(C)(C)C(=O)CCC(=O)N1CCOCC1(C)c1cn(CCN(C)C)nn1 CS(=O)c1cccc(C(=O)NC2CC2NC(=O)CCc2ccc(F)c(F)c2F)c1 C1(CCC)CN(C(C2CC(C)=NO2)=O)CCN1C(c1ccc(C(F)(F)F)nn1)=O c1(OCC(=O)NCc2cc(C)c(O)nc2)cc(F)cc(C#N)c1 Cc1oc2ncnc(O)c2c1C(=O)NCC(C)(CO)NC(c1ccncc1)=O c1(C(=O)NC2C(C)CN(C(c3c(Cl)csc3Cl)=O)C2)cc(C2CC2)cc(F)c1 c1(C(N(CCOCCCN(C(C2C(C(=O)OC)C2)=O)C)C)=O)cnccn1 Cc1cc(C)c(C(N2CCCN(C(c3cnc(S)[nH]3)=O)CC2C(C)C)=O)cc1C c1(CC(=O)N(C2CCCN(C(=O)CC3CC=CCC3)CC2)C)cc(Cl)ccc1O N1(C(C(C(C)NC(c2nccc3[nH]ccc23)=O)C)=O)CCC2C(=O)NCC2C1 C1(C(N(CCN(C(=O)CC2CCOCC2OC)CC)CC)=O)CSCC(=O)N1 C1(c2ccccc2)(CNC(=O)NCCCC2CCOC2)COCCO1 N1(C(c2nc(C)oc2)=O)CC(NC(C2CCC(=O)NC2)=O)C2(COC2)C1 Cc1ncc(NC(C2CCN(C(=O)C=CCBr)C2c2ccccc2)=O)c(C)n1 Cc1c(C(=O)NC(C)CNC(=O)Cc2ccc(Cl)cc2Cl)[nH]c2c1CCCC2 CC(CCNC(=O)C=Cc1cocn1)CCNC(=O)Cc1cccc(C(F)F)c1 c1(CC)cc(C(N2CCC(CNC(=O)CC3(O)CCCN(C)C3)C2)=O)ccc1O c1(OC)cnc(C(=O)NCCC2CN(C(=O)C(C)(C)C3CCC3)C2)c(OC)n1 CC(CC(=O)N1CC(C)(C(N2CCC(C#N)C2)=O)CC1(C)C)C(F)(F)F C(=O)(CC(C)C(F)(F)F)NC1CCN(C(C2(C=C)CCC2)=O)C1 C1(OC)CCCN(C(=O)NC2CCCN(C(c3cc(Cl)ccc3Cl)=O)C2)C1OC c1(C(=O)NCC2C=CC(NC(=O)CCC3CCC3)C2)nnc(O)c2c1CCCC2 C1(NC(c2cn(CC)nc2)=O)CCC2CN(C(c3coc(CO)c3)=O)CCC2C1 Cc1ncc(Cl)cc1C(N1CCC(NCc2cnc(O)c(Cl)c2)C(F)C1)=O c1(CC(N2CC(CCNC(=O)CC(O)CC3CC3)C2)=O)cccc2ccncc12 Nc1cccc(C(N2CCCOC(CCNC(=O)CC3CCSC3)C2)=O)c1F N1(C(c2ccncc2F)=O)CCCC2(C1)CN(C(C1CCCOC1)=O)CCO2 CC1(C)CCCC(O)(C(=O)NCC(C2CC2)NC(=O)Cc2ccccc2Cl)CC1 c1(C(N(CC(CNC(c2c(C)n(CCO)nc2)=O)O)C)=O)cc2occc2s1 c1(OC)ccc(CNC(C2(F)CCN(C(=O)C(n3cc(C)cn3)C)C2)=O)cc1C C1(NC(=O)CCc2cc[nH]n2)COC2(C1)CN(C(c1ccc(O)cc1O)=O)C2 C1(NC(c2c(C)onc2)=O)CCCCC1CNC(=O)CCCOc1cccnc1 N1(C(C2OCCC(NC(c3c(C)cncc3C)=O)C2)=O)CCC2(CCC2)CC1 c1(C(=O)NCCNC(C2(O)CCOC2)=O)cccc(C2CC2)c1F c1(SCCC)ccc(C(=O)NCC2CN(C(=O)Cc3ccc(Cl)nc3)C2)cc1 N1(C(C2C(OCC)C2C)=O)CC2CCCC2(N=c2[nH]c(Cl)c(C#N)s2)C1 C12(CNC(c3csc(Cl)n3)=O)CCC(C1)N(C(c1ccc(F)c(O)c1)=O)C2 C1(C(=O)NCC(C)NC(Cc2cc(OC)no2)=O)CCc2ccccc2CC1 N1(C(C=CCOCCOC)=O)CC2(CCCC2N(C(=O)Cc2ccsc2)CCC(C)C)C1 Cc1nc(C(C)C)sc1C(N1CCC(O)(Cn2cc(CCC(C)(C)O)nn2)C1)=O N1(C(C2C3CC4C(C3)C24)=O)CCC2(CCC2NC(c2c(C)cc(Br)cn2)=O)CC1 N1(C(C=CCC)=O)C2CCC1CC(CCNC(C1(c3ccnc(Cl)c3)CC1)=O)C2 CC1CN2CCN1C(C(=O)NC1CC1NC(=O)C(F)CC1CCCC1)C2 c1(N(C(=O)Cc2cnoc2)CC)ccc(N(C2CN(CC)C2)CCO)cc1Cl c1(C(=O)NC2CN(C(C(CC)N(CC)CC)=O)C2)cnc(C(C)C)nc1C c1(C(C)C)cc(C(=O)N(CC(O)CNC(C2(CO)CCC2)=O)C)no1 c1(NCC2N(C(c3c[nH]c4nccc-4c3)=O)CCC2)ncnc2c(Br)cccc12 C(=O)(C(C)(C)CCSC)NCCN(C(C1CCN(C(CC)=O)C1)=O)C c1(C(N(C)CC2C3CN(C(CCCC)=O)CC32)=O)cccn(C2CCC2)c1=O C1(NC(c2c(CC)scn2)=O)CC2CCC(C1)N2C(c1c(O)cccc1F)=O Cc1cc(Cl)c(F)cc1C(N1CCC(O)C(C(=O)NCc2ncccc2Cl)C1)=O C(=O)(C(F)C(=O)NCC1CN(C(=O)C(C)OCCC(C)C)CCO1)OCC c1(ONC(CN(C(C)C)C(C2CC=CC2)=O)=O)cccc(Cl)c1 c1(N2C(=O)CC(CC3CN(C(c4cn(C5CC5)nn4)=O)C3)C2)cc(Cl)cc(Cl)c1 c1(C(=O)OC)cc(Br)ncc1NC(=O)CC12COC(C)(C1)C2 c1(C(=O)NC2C(NC(C3(C)CC=CCC3)=O)COC2)cc(F)cc2cnccc12 C=CC1(CC(N2CC(CCO)(NC(c3cc(COC)on3)=O)C2)=O)CCC1 C1(O)(CNC(c2ccc(OC)cc2)=O)CCCN(C(=O)CSS(C)(=O)=O)CC1 c1(C(=O)OC)cc(C)c(NC(C2CCC(OC(F)F)CC2)=O)c(Cl)c1 S(=O)(=O)(c1ccc(N2CCC(C)(C(F)(F)F)CC2)c(F)c1)N(C(C)CC1CC1)C CCC(C(=O)NC(C1(O)CN(C(=O)Cn2cnc(C(N)=O)n2)C1)C)OC N1(C(C2(C)CC=CC2)=O)CCN(C2CCC2NC(=O)Cc2ccc(F)cc2)CC1 C(C(O)CC(=O)NCC1CCC1(F)F)NC(CCCNC(N)=O)=O c1(CC)c(C(=O)NCCOCCNC(=O)CC2CCC3CC23)csc1C N1(C(c2ccc(NC)cn2)=O)CCC(NC(=O)COc2ccccc2)C12CCC2 c1(OC)cc(C(=O)NC2CC=CCC2C(=O)NCCc2cn(C)nn2)ncn1 Cc1ccc(P(C)(C)=O)c(NC(=O)C(=O)NCC(c2cccc(F)c2)C2CC2)c1 C1(COC)CN(C(C2(C#N)CCCC2)=O)CCN1C(=O)Cn1nccc1C c1(C(=O)NCC(C)NC(CCc2cnc(C)nc2O)=O)cccc(Cl)c1[N+](=O)[O-] c1(C(=O)NC(c2cn(C3CCOC3)nn2)(C)C)cc(F)cc(S(N)(=O)=O)c1 N1(C(CC2CN(C(C)=O)C2)=O)CC(NC(C2CCOCC2)=O)CC1C C(=O)(C1=CCCN(C(c2nccn2C)=O)C1)Nc1ncc(C)cc1C C=CCC(CNC(=O)C(C)OCC)NC(c1cn(C2COC2)nn1)=O c1(C(=O)NC(C)CCNC(c2cc(F)c[nH]2)=O)cc(Br)nn1C c1(C(N(C(CNC(c2c(CC)nns2)=O)C)C)=O)cncc(F)c1Cl c1(CC)c[nH]nc1C(=O)NC1(CCNC(=O)C(C)Cc2cnn(C)c2)CC1 CC1CC(C(=O)N(C)CCN(C)C(C2COC2)=O)CO1 C1(C(=O)NCC2CCN(C(c3cc(C)c(O)nn3)=O)C2)CCC2(CCCC2)C1 c1(OC)cc(C)ccc1C(N1CC(CC(C)NC(c2csc(C)c2C)=O)C1)=O c1(C(N2CC(C)C(NC(c3cncn(C)c3=O)=O)C2)=O)ccc(F)c2ccsc12 c1(C(=O)NC2CC(NC(c3cn(CC(CC)O)nn3)=O)C2)cc2ccsc2n1C c1(OC)ccc(C(=O)NCCCCC(C)NC(c2c[nH]nc2F)=O)c(F)c1 c1(-n2cc(C3N(C(c4nnn(C(C)(C)C)n4)=O)CCOC3)nn2)ccc(Cl)c(Cl)c1 N1(C(C2CC(NC(CC)=O)C2)=O)CCCC1C1CCN(C(=O)C=CBr)C1 Cc1nc(C(N2CCSCC2CCNC(=O)CCC(C)(C)C)=O)ccc1C#N C1(CNC(C(C)C#N)=O)CC2CCC(C1)N2C(=O)CNC(=O)CCC1CCCC1 N1(C(c2cncc(C)c2)=O)CC(C)CCC1CNC(=O)CCOc1cccnc1 CC(C(C)(C)C(=O)NCC=C1CCSCC1)NC(=O)CC1CSCCO1 O=[N+]([O-])c1ccc2[nH]cc(C(COC(F)F)NC3(C4CC4)CC3)c2c1 Cc1cc(N)c(C(N2CCN(C(c3ncn(C)c3C)=O)C3CC23)=O)cc1C N1(C(c2nccc(CC(=O)OC)c2F)=O)CCNCCC1(C)C N1(Cc2cccc(C(=O)Nc3ccc(Cl)cc3F)c2)CCC2(CCOC2=O)C1 c1(C(=O)Nc2ccc(-c3cnc(OC)nc3)s2)cnc(OC)c(Cl)c1 O=C(C1CCc2scnc21)NCC1(CNC(C2COCCC2(F)F)=O)CCCC1 Cc1cc(C(=O)NCC(CNC(C2CC=CCO2)=O)CO)c2occc2c1 CC(O)C(C(=O)N1CCCC(NC(=O)CC2CCCC2(F)F)C1)N(C)C c1(COC)ncsc1C(=O)NCCCC1(CNC(=O)CC2(O)CC2)CCCC1 c1(C(=O)NCC2C(NC(c3c(CC)nco3)=O)C2)cc(Cl)cc(F)c1N C1(NC(C)Cc2ccccc2F)CN(Cc2cccc(O)c2)CC1(C)C C1(CNC(COc2c(C)cccc2)=O)CN(C(=O)C(C(C)C)NC=O)CCCO1 CC(C(=O)N1CCN(C(c2ccc(SC3CC3)cc2)=O)C(C(C)C)C1)C(F)(F)F C1(C(=O)Nc2cnc(C)nc2)CC2(CCN(C(=O)C(C)N3CC(C)C3)C2)C1 c1(C(=O)NCC2CCC(NC(C3(C)CCSCC3)=O)C2)cc(F)c(F)c(F)c1 N1(C(C(CC(=C)C)(C)C)=O)CCC2CN(C(C3CC4CCC3O4)=O)CC2C1 N1(C(c2cn(CCO)nn2)C(=O)NC2CCN(CCC)C2)CCCC(C#N)C1 C12(CNC(N3CCCC3c3cncc(Br)c3)=O)CCC(CC1)C2 C1(C(N2CC3(C(NC(CCCC#C)=O)CC3)C2)=O)CCC2(CC1)CC(OC)C2 C(C(=O)NC(C1CCN(C(c2cnc(S)[nH]2)=O)C1)(C)C)(C(C)C)NC(=O)OC C=CC(C)CC(=O)N1CCCCC1C1(NC(c2cc(C(C)(F)F)n[nH]2)=O)CC1 C1(CNC(=O)C(O)C2CC2)C2CCCC1N(C(c1cccc3ccsc13)=O)C2 c1(C(=O)NCC(CC=C)NC(=O)CC2CC(=O)NC2=O)ccc(F)c(C)c1C#N C1(C(N(C2C(C)CCC2)C)=O)(NC(=O)CC2CC=CCN2C)CCN(C)C1 CC(CCCCN=c1nc[nH]s1)NC(=O)C(C)(C)n1cccn1 c1(C(N2CC(CNC(C=C(C)Cl)=O)C(F)(F)CC2)=O)c[nH]c2c(C#N)cccc12 C1(NC(CC(n2ccc(C)n2)C)=O)CC2CCC1N(C(c1cc(C)nn1C)=O)C2 c1(OC)ccc(-c2cn(C(C)CNC3CCCN3c3ccccc3)nn2)s1 C1(CC(N2CC3C(NC(c4n(C)cc(C(N)=O)c4)=O)C3C2)=O)CCCC(C)(C)C1 C(=O)(C(CC)(CC)OC)NCCN(CCCCCC)C(c1ccnn1COC)=O c1(C(=O)NCC#CCNC(C2(c3cccnc3)CCC2)=O)ccc2cnoc2c1 N1(C(CCC(=O)NCC)=O)CCC12CN(C(=O)CCCc1ccncc1)C2 CC1(F)CN(C(C2CCCCC(=O)N2)=O)CCN(C(c2cccc(F)c2F)=O)C1 C1(CNC(C2N(C)CC(F)C2)=O)CC2(CCC2)CN1C(=O)CCNS(C)(=O)=O CC1CCCC(CC(=O)N(C2(CC(=O)NC3CC3c3cccs3)CC2)C)C1 c1(C(C)C)ccc(C(N2CC3CC3(C(=O)OC)C2)=O)cc1Br.c12cccc(n1)O2 N1(C(=O)NC(COC)C)CCCC12CN(C(c1cccc(OC3CC3)c1)=O)C2 S(=O)(=O)(c1ccccc1Cl)NCC(=O)NCC1C(c2n(CC)ncc2)OCCC1 c1(C(=O)NC(COC(C)(C)C)C(=O)O)cnc2ncnc(O)c2c1 CCC(CC(=O)N1CC(C(=O)NCCNC(C2(F)CCCC2)=O)C1)C(F)F N1(C(CN(CCC)C)=O)CC(OC)CC(NC(=O)C=C(C)c2cccnc2)C1 N(C(=NCCCF)NCCCS(C)(=O)=O)C(C(C)C)Cc1ccccc1.C1CO1 N1(C(CC(CC)SC)=O)CCC(C)(CNC(=O)C=CCN2CCOCC2)CC1 C1(C(=O)NCC2N(C(CCc3cc(C(=O)OC)[nH]c3)=O)CC2)COCCN1C c1(NC(C2(C)N(Cc3ccc(C)c(C)c3)CCC2)=O)cn2c(Br)cccc2n1 N1(C(c2c(C)nns2)=O)CC(C)C(Nc2cc(C(N)=O)ncn2)C(C)C1 c1(C(N2CC(CC)C(NC(c3cscc3OC)=O)CC2)=O)cnn2ccccc12 O=C(CCCCCO)NC1(CNC(C2CCNC2=O)=O)CCCCC1 c1(C(N(C2CCN(C(C(CC)OC)=O)C2)CCO)=O)ccc(C2CC2)cc1 N1(C(c2c(OC)n[nH]c2)=O)CCCC(C2CCCN2C(c2ccc(F)nc2)=O)C1 N1(CC)CC(NC(=O)C(=O)NCCSCCC(=O)O)OC1=O C1(c2ccc(Br)cc2)(C(=O)OC)CCN(C(=O)C(C2CCCCC2)=O)C1 C1(CNC(C2CC2C2CCC2)=O)CCCN(C(c2cc(Br)ccn2)=O)CC1 Cc1cc(O)cc(C)c1C(=O)NC1CCC1NC(C1CC1C(F)(F)F)=O C(C1CCN(C(=O)C(C)C(F)(F)F)CC1)=CC(=O)NCC(CCC)(C)O c1(C(C)=O)cn(C)nc1C(=O)NC1C2CN(C(C3CC3c3nccn3C)=O)CC12 c1(CC)c(C(=O)NC2CN(C(=O)CC3CC4CC4C3)CC2F)nnn1CC c1(C(=O)NCCNC(C2CC(C)(F)C2)=O)cccc(OC(F)(F)F)c1 C1(C(=O)NC(C2(O)CCC2)C)(COC)CCN(C(=O)C(C)OC)CC1 N1(C(C)Cc2ccc(O)cc2)CCC2(CC1)CC2C(N1CCCC(F)CC1)=O CCCC(C(=O)NCc1ccccc1CNC(C1CC1C(N)=O)=O)OCC CC(CC1CC1)C(=O)NCC1CC(O)(CNC(C2(CCF)CC2)=O)C1 C1(C)(C(N(C2(c3cc[nH]n3)CC2)C)=O)CCN(C(c2c[nH]c(=O)cn2)=O)CC1 CC1CN(C(N2CCC2C2CCOC2)=O)CCc2ccc(Cl)cc21 C(=O)(C1CNc2c(C)cccc21)N(CCC)C CN1C(=O)CSC1=C(F)C(=O)NC1COCC1NC(c1ccc2nncn2c1)=O C(=O)(CCCS(N)(=O)=O)NC1CN(C(c2cnc(SC)nc2O)=O)CC1C C1(CNC(=O)Cn2ncnn2)(CO)CC(C)(C)C1.c12ocnc1C(C)N1CC2C1 Cc1cc(C)c2[nH]c(=NC3CCCCC3CNC(=O)CCC3CCOC3)sc2c1 C1(Cn2cc(CNC(=O)OCC)nn2)CC(O)CN1C(=O)C(C)(C)C1CCOC1 C1(CCC)CN(C(=O)C=C2CCC2)CCN1C(=O)Cc1cc(C2CC2)on1 c1(C(N2C(CNC(c3nc(CCCC)sc3)=O)CC2)=O)nn(CCC)cc1Cl N1(C(c2c(C)c[nH]n2)=O)CCN(C(c2cccc(Br)c2)=O)CC1CCO Cc1nc(C(C)(C)C)[nH]c(=NC2CCC(NC(c3ccsc3C)=O)CC2)c1C C1(C(=O)NCc2snc(CC)n2)CCCCN1C(c1cccnc1C)=O C1(NC(C(F)=CCC)=O)CCC2(CC1)CC2NC(C1CCN1C(C)(C)C)=O n1(C(C)C)cc(C(C)NCC(n2cc(Br)cn2)C2CC2)cn1 C1(C(=O)NCCN2CCN(C(C(CN(C)C)N(C)C)=O)CC2)CC2(C1)CC2(F)F c12nc(c(C)cc1Br)OCCCn1c(nnn1)C2NC(CC=C)C.C1CC1 N(C(=NCCC1(O)CCC1)NC(C1CC1)C1CC1)CC1(C)C(C)CCC1 c1(C(N2CC3C(CNC(c4ccn(COC)n4)=O)(C3)C2)=O)ccc2oncc2c1 c1(CC)cc(C)ccc1NC(C1(CN(C)C(c2coc(C3CC3)n2)=O)CC1)=O CC1CCN(C(=O)CC(=O)OC(C)(C)C)C1C(N1CCC(c2ncco2)C1)=O CCC(C)(C(=O)NC1CC2CC1CN(C(c1coc(C(F)F)n1)=O)C2)C(N)=O N1(C(c2ccc(CC)cc2)=O)CCCN(C(c2cc(CSC)c(C)s2)=O)CC1 N1(C(c2ccc(Cl)c(Cl)c2)=O)CC2CCC2(C(N2CCCC(Br)C2)=O)C1 C1(C(N2C3C(CNC(C(C(C)C)(C)C)=O)C(C3)C2)=O)CC2C=CCC(C1)C2 c1(NC(CC2CCC(NC(Cc3nc(C)sc3C)=O)C2)=O)ncc(Br)nc1I C1(CNC(c2cc(SC)oc2)=O)CN(C(C2C(C)C2C)=O)C2(CCOCC2)C1 N1(C(C(C)Cc2ccco2)=O)CC(F)CC1CNC(=O)Cn1ncccc1=O CC1CC(c2ccccc2)(C(=O)NC2CCC(NC(=O)CCC3OCCO3)C2)C1 C(=O)(C(C)N(OC)C(=O)C(C)c1cc(C)cc(C)c1)OCC c1(C(=O)NC(C2CN(Cc3c(C)nccc3)C2)C)ccc2c(c1)NC(=O)CO2 c1(C(C)C)ccccc1C(F)(F)C(=O)NCCc1nc[nH]n1 N1(C(C(C)OCC(C)C)=O)CCOC2(CCN(C(=O)C(C)NS(C)(=O)=O)CC2)C1 Cc1ccc2[nH]c(CNc3[nH]cnc3C(N)=O)cc2c1.N12CC(CC(F)C1)C2=O C1(F)(C(=O)NCCN(C(C)C)C(=O)CC2NC(=O)NC2=O)CCN(C)CC1 c1(OC)ccccc1C.CCS(=O)(=O)NCC(=O)OCCN(C(=O)CCOCC)C C1(C)(CC)CCN(C(C2(CNC(=O)CSCCC(C)C)CCCC2)=O)C1 n1(CC)ncc2cc(C(=O)N(C)CC3(OC)CCOC3)cnc12 C1(NC(c2[nH]cc(C)c(=O)c2)=O)CN(C(=O)C(F)C(F)(F)F)C2(CCC2)C1 c1(C(=O)O)ccc(CC(CO)NC(C2CC2c2ccsc2)=O)cc1 C1(CNC(c2c[nH]cc2Br)=O)CC2CN(C(C3(F)CCCCC3)=O)CC12 C1(NC(c2cc(CF)on2)=O)CN(C(C2C3CCCOC23)=O)CC1C(F)(F)F c1(C(C)NC(c2ccc(CNC)s2)=O)cnc(C(F)(F)F)c(OC)c1 C(C(=O)NCCCCC(=O)NCc1csc(C)n1)(C(C)C)OC c1(NC(c2c(CC)nn(C)c2)=O)ccc(NC(=O)C(C)(C)COC(C)C)c(C)c1 N1(C(CCc2c(C)ncs2)=O)CC(NC(=O)CCS(=O)(=O)N(C)C)CC1(C)C C(CCC(O)C(=O)NCC1CCC1)NC(C1C(C)(C)C1(F)F)=O Cc1nc(C(=O)NCC2(C(N3CCC3CN(C)C)=O)CC2)cn1C c1(C(N2CCN(C(C(NOC)=O)=O)C(CO)C2)=O)c(C)cc(C)nc1S S(=O)(=O)(c1ccc(C)cc1F)Nc1scc(C(=O)NCC(CC)OC)n1 C(=O)(C1=CC2(CCOCC2)C1)N1CC(OC)C(NC(c2nc(Cl)sc2C)=O)C1 C1(NC(=O)CCc2cccc(O)n2)CCCCCN(C(=O)CNC(=O)C2CC2)C1 C(CC(CC)C(=O)NCC(O)CN(C)C(C1CCN1C1CCCC1)=O)=CC C(=O)(CCC(C)(C)c1ccccc1)NC1(CF)CCN(C(COC)=O)C1 c1(C(c2ccccc2)COC(C)=O)ccc2c(c1)OCO2.C1(C(C)C)C(=O)N1 c1(OC)cccc(OC)c1CC(N1CCN(C(C2CC2F)=O)CC1CC(F)F)=O CCC(C)CC(=O)C(=O)N1CCC2(CC1)CC2C(N1CC(C)(C)CC1C)=O C(=O)(C=CS(C)(=O)=O)NCC(C(C)C)NC(=O)Cc1ccccc1Cl c1(C(N2C(CN(C(CCOCC(C)C)=O)C)CCC2)=O)cccnc1S N1(C(CCC=CC)=O)CCCC2CN(C(c3ccc(F)cc3O)=O)CCCC12 N1(C(C(c2ccc(C)o2)C)=O)CCC2(C=C(C(=O)NCc3nccn3C)C2)C1 C1(C(=O)NCC(CC)(C)Cl)CN(C(=O)Cn2cnnn2)CC12CCC2 N1(C(Cc2n[nH]c(=NC)s2)=O)CC(NC(c2cnc(OC)cc2C)=O)C(C2CC2)C1 c1(C(=O)Nc2cc(C)c(F)cn2)ccc2c(c1)CCN(Cc1c[nH]ccc1=N)C2 N1(C(C(n2c(C)cc(C)n2)C)=O)CCOCC(NC(=O)C=CSCc2ccco2)C1 C1(C(C)(C)C(=O)NCCOC(=N)O)CCCN(C(=O)COCC2CC2)C1 O=C(CC1COc2ccccc21)NCC1CCN1C(c1cccn2nccc12)=O CC1C(C(=O)NC2CCC3CCC23)CCN1C(=O)CC1CCCC(=O)C1 C1(NC(CCc2cc(C)on2)=O)CN(C(=O)C=CS(C)=O)CC1CC(C)(C)C c1(C(N2CC(N(C)C(C3CCCOC3)=O)C2)=O)ncc(OC(C)C)cn1 c1(C(N(C(c2cn(-c3ccnc(F)c3)nn2)C)C)=O)ccc2c(c1)OCC2 N1(C(C=CC(N)=O)=O)CCC2(C1)c1[nH]cnc1CCN2C(=O)CC1CCNC1=O N1(C(CC2N(C)CCOC2)=O)CCC2CCC(NC(c3ccc(F)cc3N)=O)C12 C1(C(N2C(Cc3ccc(C)cc3)(CO)CC2)=O)CN(C)C(=O)CN1 C(c1ccc(C(=O)O)o1)=CC(=O)N(CCC(=O)O)CCc1ccccc1 C1(CC(N2CC(N(C(c3n(CC)ncc3Cl)=O)C)C2)=O)CCCNC(=O)C1 C#CCC(C(=O)N1CCCC1C=Cc1cccs1)NC(=O)OC(C)(C)C C(=O)(C(CC1CCOCC1)NC(=O)COCC(F)F)N(C1CC(OC)C1)C c1(CC)cc(C(=O)NC2(CNC(=O)CCc3scnc3C)CCC2)ccc1C C=CCC(C(=O)N1CCCC1(C(=O)NCC(O)CC1CCCC1)C(C)C)OC C(=O)(CCCCCO)N1CCC(CNC(CCC(C)OCC)=O)C1C C1(O)(C(N(CCCNC(C2(CCOCC)CCCC2)=O)C)=O)CCCC(C)CC1 CC1(C)CC(Nc2cnn(C3CCNC3)c2)Cc2ccccc21 C1(F)(CNC(COC(CC(C)C)C)=O)CCC(NC(=O)C(C2CCC2)C2CC2)C1 C1(N(C(=O)CC2CCS(=O)(=O)C2)C)CC2CN(c3ncc(Br)c(O)n3)CC2C1 C1(C)(CNC(C2CN(C)C(=O)C2)=O)CN(C(C2(C)CCC3CC3C2)=O)CCO1 c1(CCC)nc(C(=O)NCC2(NC(=O)C(F)n3cccn3)CC2)co1 C12(C(=O)NCC(C)NC(Cc3c(C)ocn3)=O)CCCCCC1OCC2 C1(C(=O)NCC2(CNC(c3coc(Cl)n3)=O)CC(F)(F)C2)Cc2ccccc2C1 C(=O)(C(C)(C)CC(=O)NCC1(O)CCCN(C(C2C=CC(=O)N=N2)=O)C1)OC N1(C(CS(CC)=O)=O)CC2(CCCC(CNC(c3cc([N+](=O)[O-])c(C)s3)=O)O2)C1 CC(C)C(F)(CNC(=O)C(C)C1(O)CCC1)C(=O)NCC1(C)CC1(F)F N1(CC(CC)C)CCCC(C(=O)Nc2csc(C)n2)C1 C12(NC(CSC)=O)CCN(C(c3cccc(N)c3Br)=O)CC1C2 N1(C(c2c(C)cc(Br)cn2)=O)CC2CCN(C(c3n[nH]cc3F)=O)CC12 CCCCCC(O)C(=O)NCCNC(c1cccc(C2CNC(=O)C2)c1)=O Cc1cn2c(n1)CC(C(=O)NC1CC(CNC(C3(C)CCCCNC3=O)=O)C1)C2 C1(C(N(CCCCCNC(C=C(C)C)=O)C)=O)CCCC12CC2 C1(O)(c2cn(CC(CC)O)nn2)CCN(C(c2ccc(COC)c(F)c2)=O)CC1 c1(CNC2CCC(C(=O)NC(C3CCOC3)C)C2)ccc2c(c1)CCCO2 c1(CC)oncc1C(c1nnnn1Cc1cccs1)NC1CCCCC1 C(=O)(CC1=CCN(C(=O)CCCC#C)CC1)NC(C#C)C(C)(C)C c1(C(=O)NC2CC(C)(CNC(C=C(C)C)=O)C2)ccnc(Br)c1N C1(n2c(-c3cc(Cl)c[nH]3)nc(C(CCC)C)n2)CC(C)(C)OC1(C)C N1(C(Cc2ccc(OCC)cc2)=O)CC2CC(C)N(C(=O)C(C)CC(F)F)C2C1 C1(CC)C(NC(C2COCCC2(F)F)=O)CCCN1C(c1sccc1C)=O c1(C(=O)NC(CCN(C(C(C)NC(=O)NC)=O)C)C)cncc(-n2ccnc2)n1 CC1CN(C(=O)C=C2CCC2)C(C)CN1C(c1cccc(OC(F)F)c1)=O c1(NC2CC(O)(CNC(C3CC=C(C)CC3)=O)C2)ncc2ccnc-2[nH]1 C1(C(=O)NCC=CCC(=O)NCC(C)OCC#C)CCCCCC1 c1(CNC(C2N(C(c3ccc(C)cc3)=O)CCC2)=O)cc2c(nc1O)CCOC2 c1(OC)cccc(OC)c1C(=O)NC(C)CCN(C)C(C1(C)CCNC(=O)C1)=O C=CC1(O)CCN(C(=O)C(CCNC(c2cncc(NC)c2)=O)OC)C1 C(=O)(C1=NN(CCO)C(=O)CC1)N1CCC(F)(CNC(C23CC4CC2C3C4)=O)C1 c1(C(N2C(CNC(c3ccc(=N)[nH]n3)=O)CCC2)=O)cc2cc(F)c(Cl)cc2[nH]1 C=CCC(CNC(C1C(O)CCN1C(c1ocnc1CC)=O)=O)CC(C)C C1(CO)CN(N2CCOC(C)(C(F)F)C2)C2(CCCC2)C1 Cc1ccc(Br)cc1C(=O)N(C)CC1CCCCN1C(C1CCC(=O)O1)=O Cn1cc(C(N2CCC(CO)(CNC(=O)C(F)C3CCC3)CC2)=O)c(O)nc1=O c1(C(N2CC(COC)N(C(=O)C(C)CN(C)C)CC2)=O)ccc2cncn2c1C c1(NC(C(C2CC(C)OC(C)C2)F)=O)cc(F)c(N)c(F)c1F c1(NCC2(NC(Cc3cccc(CC)c3)=O)CCC2)ncnc2cc(C)[nH]c12 c1(C(C)NC(CSCCNC(C(C)OCCC=C)=O)=O)ccc(O)cc1 c1(CNC(N2CC3(C(C(N4CCCC4)=O)C3)C2)=O)cc(F)ccc1Br CC(CN1CCCCC1)C(=O)NCC1CC(CNC(=O)C(C)(Cl)Cl)CO1 c1(C(N(C2CCC(NC(c3ccc(CCC)[nH]3)=O)CC2)C)=O)cccc(N)c1C c1(CCCC(=O)N2CC(C(C)NC(=O)C=CC3CCOC3)C2)ccc(F)cc1 c1(CC(=O)NCCCOCCC(=O)NC(c2ccccc2F)C)cccnc1O c1(-c2nc(C)sc2)cccc(C(=O)N(CCC#N)CC2CC2)c1 c1(OC)ccncc1C(N1CCC(OCCNC(=O)N(C)C)C1)=O c1(N2CCC3(CC(NC(C(CC)OC)=O)C3)C2)c(Cl)cccc1[N+](=O)[O-] C1(O)(CC#C)CC(C(=O)NCC#CC(=O)NCCCC=CC)C1 C1(CCC)CN(C(=O)CC2CC3CC3C2)CC1C(N1CCCC1CC(C)C)=O c1(C(=O)NC2C(NC(C(C)(C)OC)=O)CCC2)c[nH]c2ccc(I)cc12 CC1CN(C(=O)CCN(C)C(=O)NCc2nocc2Br)CC(C)O1 Cc1cc(C)c(C(N2CC(C)C(F)(F)C2)C(=O)NCCCF)c(C)c1 c1(C(C)C)nocc1C(=O)NCCN(C(=O)CC1CCCN1C(C)=O)C.C(C)(C)(C)O C1(CC)CN(C(=O)C(C2CC2)SC)CC1C(N1CC(COC)(OC)C1)=O C1(NC(CN(C(C)C)C)=O)CC2(CCC(CNC(=O)C(F)C3CCCC3)OC2)C1 C1(C(=O)OCC)(COC)CCCNC1.N12CCN(CC1)C(=O)NCC2 N1(C(C(c2ccc(F)cc2)C)=O)CC2CC1CC2CNC(C1CN(C)C1)=O C(=O)(CS(=O)(=O)C1CC1)NC1CC(C(C(N2CC(C)C(C(N)=O)CC2)=O)F)C1 Cc1cc(C(N2CCN(C(c3ncon3)=O)C(CO)C2)=O)cc(C#N)c1 N1(C(CN(CC)CC)=O)CCCCC1C(C)NC(c1ccc[n+]([O-])c1)=O C1(CN(C(C2CCC(C)C2)=O)C)CCCCN1C(c1coc(Br)c1)=O N(C(=NCc1ccccc1)NCc1cc(C)ns1)CC(CC)CO c1(CCN(C)C(=O)NCc2noc(C3(C)CCCC3)n2)nccc(O)n1 N1(C(CSC(C)C)=O)CCC(C(C)NC(=O)Cc2cc[nH]n2)CC1 C1(CNC(CNC(CC)=O)=O)CN(C(=O)C(C)N(C)C)CCC1(C)C C1(N(c2ccc(C(C)C)cc2)C(c2cccnc2S)=O)CC2CCC(C1)N2 N1(C(C2C=CCN(C(Cc3scc(C)c3)=O)C2)=O)CCCN(C2CC2)CC1 C(=O)(C(O)CC(C)(C)C)NC1C2CN(C(Cc3cccc(C(C)C)c3)=O)CC21 C1(C(N2CCCC(NC(c3ccc(O)cc3)=O)C2)=O)(OC)CCSCC1 c1(CC(=O)NCC2CC(O)(CNC(C(C)(C)OCC)=O)C2)cc(F)c(C)cc1F N1(C(C(COC)O)=O)CC2CCC1C1CN(C(c3cscc3SC)=O)CC21 N1(C(C=C(CC)C)=O)CCC2(CCCCC2NC(c2nc(C3CC3)oc2C)=O)C1 c1(C(=O)NCC(CNC(c2c(C)c[nH]n2)=O)(C)C)ccc2c(c1)C(C)CN2 c1(C(=O)NC2(CN(C)C(c3nccnc3N)=O)CC2)ccc(C(F)(F)F)c(Cl)c1 c1(C(=O)NC2CN(C(c3cc(OC)n[nH]3)=O)CC(O)C2)n[nH]c2c1CCCCC2 C1(NC(c2ccc(C)c(F)c2N)=O)CCN(C(C2CC=CCC2)=O)CC12CCC2 c1(OCC)cc(Cl)ccc1C(N1CC2CC2(NC(C2C=CCC2)=O)C1)=O c1(OC)cc(Cl)ccc1-c1ncc(C)s1.c12ccc(cn1)CN(CCO)CC2 C#CCC(C)C(=O)N1CCC(NC(c2c(C)nsc2OC(C2CCCC2)=O)=O)C1 C1(NC(C(C)(C)NC(C)=O)=O)CC(O)CN(C(c2cc(C(=O)O)c(F)cn2)=O)C1 C(c1ccncc1)=C(C(=O)NCC(CC)NC(C1CCN1C)=O)C N1(C(C(F)=CCC)=O)CC2(C1)CN(C(C1(c3cncs3)CC1)=O)CC2CO c1(C(=O)NC2(n3cc(CCCO)nn3)CC2)conc1C(F)(F)F Cc1ccccc1C(C)(C)NC(=O)C(=O)NCCCNC(N)=O CN=c1nc(N2CCC(C3CCCO3)CC2)[nH]c(=NCc2ccnnc2)[nH]1 c1(C(O)CN2CCN(c3cc(C4CC4)[nH]n3)CC2)ccc(Cl)c(Cl)c1 c1(C(N2CC3C(NC(C4(c5ccc(OC)cc5)CC4)=O)C3C2)=O)nccc(Cl)c1O CC(C)(C)C(C#N)C(=O)N1CCN(C(=O)C(C2CC2)C2CC2)CC1CF C(CC(C)C(=O)NC(C(=O)NCc1cnn(CCO)c1)C1CCCO1)=CCC c1(NCC(c2nccs2)C)nc(N(C)CC2CCOC2)nc2c1ncn2C Cc1cc(C(=O)NCCC(C)(C)NC(c2nnc(S)n2C)=O)ccc1C(F)(F)F Cc1ccc([N+](=O)[O-])c(NC(C2(F)CCN(Cc3ccc(Br)o3)C2)=O)c1C C1(NC(=O)COC2CCN(C(c3cn[nH]c3)=O)C2)CCC2(CCC2)C1 N1(C(C2C(C(C)C)C2)=O)CC(C(=O)NOCC(C)O)CC12CCC2 C1(CC)CCOCCN1C(C1CCC(C(F)(F)F)CC1)=O C1(C(=O)NC2C3CN(C(c4c(SC)csc4)=O)CC32)CCn2c(cnc2C)C1 c1(NC(=O)Nc2c(S(C)(=O)=O)csc2)cnc2c(c1)C(=O)NCC2 C(=O)(C(C)CCC(C)(C)C)N1C(C(N(CC=C)CCOC)=O)COCC1 C1(C(N2CC3C(CNC(c4c(C)nccc4Cl)=O)(C3)C2)=O)CC2(CCCC2)CO1 c1(C(N2CCN(C(CCC(=O)NC)=O)C3C2C3)=O)nnn2cc(C)nc(O)c12 c1(CCC(=O)NCCC2CC(NC(C3(CC)CCCC3)=O)C2)nnc(C)n1C Cc1ccn2ncc(C(=O)NC(C)CN(C)C(c3ccc(C)c(Cl)c3N)=O)c2c1 c1(C(=O)OCC(=O)NCc2n(C)ncn2)ccc(CCN2CCOC2=O)cc1 c1(C(N2CCCCC2NC(=O)OC(C)(C)C)C(=O)NCC)ccc(C)c(C)c1C Cc1cc(Br)ccc1CC(N1CCC(CN(C)C(c2ccoc2Cl)=O)C1)=O N1(C(c2nc(C)sc2C)=O)CCC2CCCN(C(=O)Cn3nccc3C)C2C1 c1(NC(C2CCCC(NC(C=CCOC)=O)CC2)=O)ccc2c[nH]nc2c1 C1(C)(CNC(c2c(OCC)scc2)=O)CCN(C(C23CC(CN2C2CC2)C3)=O)C1 c1(CC)cccc(C(=O)NCC(O)CNC(C2(COC)CCOC2)=O)c1 C(=O)(C(C)(C)C(N)=O)NCCOCCN(C(CN(C)C(N)=O)=O)C N1(C(c2ccc(C3CNC3)cc2)=O)CCCC(C2(O)CC2)C1 N1(C(=O)CCn2ccnc2)CCC2(CCCN2C(c2ccccc2CO)=O)C1 Cc1csc(=O)n1CCC(=O)NCC(C1CCC1)NC(C1CC=CCO1)=O C1(NC(c2c(-c3cn(CC)nc3)n[nH]c2)=O)COc2ccc(Cl)cc2O1 C1(O)(CC#C)CCN(C(C2CCN(C(c3cc(Cl)n(C)n3)=O)C2CC)=O)CC1 N1(C(C(N2CCN(C(=O)CN3CCCC3)CC2)C)=O)CC2CCCC1CCC2 C(CNC(c1ncc(C)cn1)=O)(CC(F)(F)F)NC(CCC(=C)Cl)=O N1(CC(N2CC(OCC(=O)N(CC(F)F)CCC)C2)=O)CCCCC(=O)C1 C(N=c1[nH]c(=NCCc2cocn2)[nH]c2c1CC(C)CC2)c1c(C)nns1 N1(C(CCC2C(C)C2)=O)CC(CNC(=O)CC2(N(C)C)CC2)C2(CCC2)C1 Cn1c(O)nc(NCC2CCN(C(c3csnc3Cl)=O)C2)cc1=O c1(C(C(=O)OCC)NC(=O)CC(N)Cc2ccc(Br)cc2)cc(F)cc(Cl)c1 N1(C(CC2N(C(C(CCC(C)C)=O)=O)CC3(CC3)C2)=O)CCC(C)C2(CCC2)C1 N1(C(c2cnc(SC)s2)=O)CCC(NC(=O)OCC(C)(C)C)CC1 C1(C(N(C)C)=O)C2CN(C(=O)C(c3cscn3)NC(=O)OC(C)(C)C)CC12 N1(C(C2CC(C)C2)=O)CC2(CCCCN(C(c3cocc3Br)=O)C2)C1 N1(C(c2c(C)csn2)=O)CC(C2CN(C(c3cc(Cl)nn3C)=O)C2)C1 Cc1ccc(C(=O)NCCC2(NC(=O)CC(O)C(C)C)CC2)c(Cl)c1Cl Cc1ccc(F)c2oc(C(=O)NCC3CCCN(C(C4OCCCO4)=O)C3)cc12 Cn1nnc2c1CC(C(N1CC(NC(C3(C)COC(C)(C)OC3)=O)C1)=O)CC2 N1(C(C2C(C(=O)OC)C2)=O)CCC2(CCCN(c3ncc(C(C)(C)O)cn3)C2)C1 S(=O)(=O)(c1cccc(C#N)c1Cl)NC1CC(CNC(=O)OC(C)(C)C)OC1 N1(C(CC2C(NC(=O)C(O)C3CC3)CC2O)=O)CCCC(CF)C1 N1(C(CC(=O)NCC#C)=O)CCCC(C)(CNC(c2cc(C(N)=O)ccn2)=O)C1 c1(C(=O)NC2(C)CC(NC(C(C(CC)C)O)=O)C2)ccc([N+](=O)[O-])nc1 N1(C(CCC#C)=O)CC(CNC(c2cccc(N(C)C)n2)=O)OC2CCCC12 Cc1nnc2n1CC(C(=O)NC1CCN(C(=O)C(C)C(O)C(C)C)CC1)N(C)C2 C1(C(N2CCC(NC(CC(COC)COC)=O)C2)=O)CCc2[nH]nc(O)c2C1 c1(CC(C2CC2)Nc2cc(CO)ncc2)ccc(F)cc1F CC1CCN(C(=O)CC2CCCCC2O)CC1CNC(C1(NC(N)=O)CC1)=O c1(-c2cccn(C)c2=O)cnc2[nH]cc(C(=O)Nc3ccccn3)c2c1 C1(CC=C)(NC(=O)C(O)C(C)C)CCN(C(=O)CC2CC2C)CC1 C(=O)(C(C)S(N)(=O)=O)NCC1(C)N(c2cc(C(=O)OC)ncn2)CCC1 C1(NC(C2(C)COCCO2)=O)CC2CCC1C1CN(C(=O)CCCN=[N+]=[N-])CC21 c1(C(N2CC(CC(C(=O)NCC3(O)CCC(C)C3)F)C2)=O)ccc(O)cc1F C(CCCC(=O)NCC(C)NC(C1CC1(F)C(=O)OC)=O)NC C(c1ccc([N+](=O)[O-])cc1)=CC(N1CCCC(NC(C2(COC)CC2)=O)C1)=O c1(CCNC(c2ccc(NC(=O)OC(C)(C)C)cc2)=O)ccc(Br)c(Cl)c1 c1(CN2CCCC(C(N3CCOC(C)C3(C)C)=O)C2)cccc2c1OC(F)(F)O2 c1(C(CC)C)nccc(=NCCN(C(=O)CNC(=O)N(C)C)CC)[nH]1 CC#CCC(C(=O)NCC1(C)CC(O)C1)NC(=O)CCN(CC)CC N#Cc1cc(CN2CC(C(=O)Nc3cc(F)cnc3Br)C2)ccc1O c1(OC)ccc(C(=O)NCC(C)(C)NC(=O)CC(C)OC)c(OC)c1C N1(C(C2C(C)OCCO2)=O)CCC(F)(CNC(=O)CC2CCCC2)CC1 N1(C(CC(C)c2ccncc2)=O)CCC2CN(C(c3cncc(N)n3)=O)CC12 C1(CC)(NC(c2cn3ccsc3n2)=O)CCCN(C(C2CC23CCCC3)=O)C1 c1(C(=O)NC2CC(C)CN(C(=O)C=C3CCN(C)C3)C2)nccc2c1CNC2=O c1(C(=O)N(C)CCOC)ccc(NC(=O)NCCOCCC=C)cc1 C1(C)(OC)CN(CC(N2CC(O)(C(F)C(N3CCC(N(C)C)C3)=O)C2)=O)C1 CCC(C)(O)C(=O)NCC(F)CNC(=O)CCc1cnc(C)s1 c1(OCC(=O)NC2CC3(C2)CC(CF)C3)ccc(Cl)c(F)c1 C1(NC(c2cnc(SC)nc2)=O)CN(c2nc(SC)ncc2C#N)CC(F)(F)C1 C=CC1COCC1NC(C1CC(NC(C2(CC)CCCCC2)=O)CCO1)=O Cc1c(C(=O)NCCC2CC(C(=O)NCC3CC4(CCC4O)C3)C2)c[nH]c1C#N C(CCC(C)(C)C(=O)N(C1CN(C(C)=O)C1)C)NC(C(C(=O)OC)C)=O C(=O)(CN=c1[nH]c(C)cs1)N(CCCCNC(C=CC=CCC)=O)C N1(C(c2ccc(C)nn2)=O)CCN(C(=O)CC2CN(C)C2)CC1C1CCCC1 c1(C(CNC(C2(OC)CC2)=O)NC(c2cnn(C)c2)=O)cccc(Cl)c1Cl N1(C(=O)COC(F)F)CC2CS(=O)(=O)CC2(NC(C2(F)CCCCC2)=O)C1 Cc1nc(F)ccc1NC(=O)CC1CCCCC1NC(C1CCCS1)=O c1(N2CCC(NC(c3c(COC)scc3)=O)(CF)C2)ncc2ncn(C)c2n1 C(C)(CCC(C)C)(c1n(CCOC)nnn1)N(C(C)C)CC1CCCO1 c1(C(N(C2CC(NC(c3ccc(N)cc3O)=O)C2)C)=O)cccc2c1CCC2 C(c1ccccc1)=C(C)C(=O)NC(C1C(C(=O)N(C2CC(O)C2)C)C1)C c1(C(C(=O)NC(CNC(c2c(C(N)=O)cccc2)=O)CO)O)ccc(F)c(Cl)c1 C1(F)(CNC(C(C)OCCC#C)=O)CC(NC(=O)C(C)SCCCC)C1 C1(CC)(OC)CN(C(C2(CNC(=O)CN(C)C(C)=O)CC2)=O)C1 C(C(=O)NOCCC1CC1)(C(C)(C)C)NC(C(C1CCC1)OC)=O C(=O)(C(C)(F)C(=O)N1CCN(CCCNC(=O)C(C)(C)OC)CC1)OC c1(N(c2nnc(C(F)F)n2CC(=O)N(C2CC2)CC2CC2)C)c(C)nn(C)c1C Cc1nc(CCC(N2CC(O)(CNC(c3cnoc3-c3cccs3)=O)C2)=O)n[nH]1 c1(C(N2CCN(CCCCOC)C(C)(C)C2)=O)ccccc1N=c1ccn(C)[nH]1 c1(S(c2c(C)cc(C(F)(F)F)nc2)(=O)=O)cccc(N=S2(=O)CCCC2)c1 c1(NC2(CNCc3cncc(N(CC)CC)c3)COC2)c[nH]c2nccc(Cl)c12 CC(CC(=O)NCCN(CCO)C1CC1)C1CCCC1.O(C(F)F)CCO C#CCCN=c1scc(-c2ccc3c(Br)c[nH]c3c2)n1CC(CC)OC C1(C(N(CCC)CCNC(C2CCCC(OC)C2)=O)=O)CC2(C1)OCCO2 N1(C(c2[nH]cc(C)c2)=O)CCN(C(=O)Cc2csc(NC=O)n2)C2COCC12 C1(NC(c2cncc(C)c2)=O)CC(C(=O)NCC2CCSC2)=CC1O C(=O)(C1=NOCC1)NC1C(NC(CNC(C2CCCC2)=O)=O)CC1 c1(N(C)Cc2onc(CCC(C)C)n2)cc(I)c(Br)cn1 c1(OC)ccc(C(N2CC(OCCNC(=O)CCC(C)SC)C2)=O)cc1Br N1(C(C(=O)NC2CCN(C(c3ccc(Cl)cc3)=O)CC2)=O)CCC2C(O)CC12 CC(C)CC(C)(C)C(=O)NCC(F)CNC(c1cc2occc2n1C)=O C1(C(=O)NC2CC(C)(NC(c3nc(OC)oc3)=O)C2)C2CCC1(C)C2(C)C Cn1ncc(S(C)(=O)=O)c1C(=O)Nc1ccc(Br)cn1 C1(CNC(c2cncc(OC(C)C)c2)=O)CCN(C(=O)CC2CCCO2)C12CC2 N1(C(C2N(Cc3c(C)nc[nH]3)CCOC2)=O)C2COCC1CC(F)C2 C12(C(=O)NC3CC4CN(C(C5CN(CC)C(=O)C5)=O)CC43)CCC(CC1)C2(C)C N1(C(C(C2(O)CCCCC2)NC(C(C)OCC)=O)=O)Cc2ncsc2C1 Cc1nn(C)c(C)c1C(N1CCC1CNC(=O)C(O)CN1CCCC1)=O c1(NC(C)C)ccc(C(=O)NC2CCCC2NC(c2ccc(C(N)=O)s2)=O)cn1 C(=O)(C1CCCc2scnc21)N(CCCCCNC(c1cccc(SC)c1)=O)C N(C(=NCC)NCC1CCCC(C)O1)CC(C=C)(F)F c1(C(=O)NCC(C(=O)N(C(C)C(C)SC)C)OC)ccnnc1O N1(C(c2csc(N3CCCCC3)n2)=O)CCNC(C(N2CCCC2)=O)C1 O=C(N=c1[nH]ccc2cc(Br)ccc12)C1CSCCN1C(=O)C(F)F CCN=c1[nH]c(C)c(C(=O)NCC(O)CNC(c2cc(C)nc(C(F)F)n2)=O)s1 CCC(CCC(=O)NCc1cc(C(N2CCCC2C2CCCC2)=O)ccn1)OC Cc1ccc(F)cc1NC(C1CCC(C)CN1C(=O)C(C)CC1CC1)=O N1(C(C2C(=C)C2)=O)CCOC2(CCN(C(c3cc(Cl)ncc3F)=O)C2)C1 C(=O)(CCC(C)(C)F)NC1CC(CC(=O)NCC2(OC)CCCCC2)C1(C)C c1(C(=O)NC2C(NC(Cc3c(C)noc3Cl)=O)C2)cccc(Cl)c1O CC1(NC(c2cnsn2)=O)CCC(NC(C2CC(N3CCCC3)C2)=O)CC1 N1(C(C2ON=C(CC)C2)=O)CC(NC(=O)Cc2sc(C)nc2C)C2(CC2)C1 c1(OC)cccc(C(=O)NCC(c2ccccc2)CNC(=O)CC(C)C)c1F S(=O)(=O)(c1ccc(C)c(Cl)c1)NCC1CCN(C(C=C(C)C)=O)CC1(F)F C1(CC(N2CC(C(C)NC(C3(F)CCC3)=O)OCC2)=O)CC2CCC1CC2 Cc1cc(C(=O)NCC2CC2NC(=O)C(C)CC(C)C)cc2ccoc12 N1(C(C(CSC)OC)=O)CC2(C1)CN(C(c1cccc(F)c1Br)=O)C2 CC(CNC(=O)CN1CCSCC1)CC(=O)NCCC(O)C(F)F O=C(C(F)C1=CCCCC1)NC1CCc2ncccc2C1 c1(-c2nc3nn2-3)ccnc(Cl)c1OC.c1(CCC)ccc(Cn2cccn2)cc1 c1(-c2cccc(-c3n(C(c4cnccn4)C)ccn3)c2)cc[nH]c2nccc1-2 N1(C(c2nc(C(C)NC(CCCCC(C)C)=O)oc2)=O)CC(C)(C)C2COCC12 CN1CC=CCC1CC(=O)NCC1(NC(=O)C=Cc2ccccn2)CCOC1 C(=O)(CCCC(C)(F)F)NC(CC(C)NC(=O)Cc1cncc(C#N)c1)C CC1OC2(C)CC1(C(N1CC(NC(c3cccc(F)c3)=O)C(O)C1)=O)C2 C1(OC)CC2CC(C(=O)NC3CCC(NC(c4cc(C(C)=O)cs4)=O)CC3)CC12 c1(N2C(CNC(CN(CCOC)C)=O)CC3(CC3)C2)ccc2c(n1)CCCC2=O N1(C(c2ncn(C)n2)=O)CCC2(CC1)CC2(CO)CNC(=O)CNC(=O)C1CC1 C1(NC(c2c(C)n[nH]c2)=O)(CNC(c2cc(C)n(C)n2)=O)CCC(F)(F)CC1 c1(C(N2CCC(C)(CNC(C3CCCC(C)(C)O3)=O)C2)=O)ccn2nccc2n1 C12(NC(CC(C=C)C)=O)CCCC1(F)CN(C(=O)CCC=CC)C2 c1(C(=O)Nc2cc(C(=O)OC)c(Br)cc2C)cccc2nn(C)nc12 n1(CC)nc(C(=O)NC(C2CCN(C(C)=O)CC2)C)cc1O.C12(CC1)C(=O)NC2 CCCC(C(O)C(=O)NCC(C)O)NC(C1CCCCS1)=O C1(CCNC(C2C(C)C2C)=O)CSCCN1C(=O)COC(C)(C)C(F)(F)F CON(CC1CC1)C(=O)CNc1ccsc1C.C12CCCC1C(=O)N2CC N1(C(c2c(C)occ2)=O)CCN(C(=O)COC2CCOC2)CC2(C)CCCC12 C(c1sc(Cl)nc1Cl)=CC(=O)NC1C(OC)CN(C(c2ccncn2)=O)C1 c1(OC)cc(C(=O)NCCC2(NC(=O)C(n3ccc(C)n3)C)CCCC2)n(C)n1 c1(CNC(=O)NCC(c2ccc(F)cc2Cl)C(F)F)cnc2nccn2c1 c1(C(=O)NCC2CCC(NC(c3cc(C#N)on3)=O)CC2)c(F)cccc1Br C1(O)(CNC(=O)CC(CC2CC2)NC(=O)CC2C=CCCC2)CC2CCC1O2 c1(C(N2CCC(CC(=O)OC)C2)=O)cccc2c1CNCCO2 Cc1nc[nH]c1CC(=O)NCC(C)N(C)C(c1ccc(CC2CC2)s1)=O c1(CC(=O)CNCC(Cl)=CCl)ccc(Cl)cc1Cl N1(C(=O)Cc2ccc(F)cc2)CCCN(C(C2CCSC2)=O)CC1 N1(C(C2CCOC2=O)C(=O)NC)CCOCC1c1ncnn1C C1(NCCc2ccc(C)c(C)c2)CCCC(F)(F)CC1 c1(C(=O)OCC)nc(C(N2CCOC(c3nncn3C)C2)=O)c(C)s1 C1(N(C(=O)Cn2cccn2)C)C2CN(C(C3CC4CC3C4)=O)CC12 CCCC(O)CC(=O)N1CC(NC(=O)Cc2ccnc(O)c2Br)CC(F)C1 c1(C(=O)NC2CCN(Cc3ccc(OC)c(Cl)n3)CC2F)cc2n(n1)CCNC2 N1(C(CC2OCCN(C(c3cc(C)sc3)=O)C2)=O)CCC(CO)C(O)C1 c1(OC(C(C2CC23CCCC3)N(c2ccccc2C)CCC)=O)ccc(C)cc1 C1(OC)CN(C(=O)COC(F)F)CC1NC(c1ccc(-c2cccs2)s1)=O C1(CNC(CCCC)=O)CC2(CCN(C(=O)C3=C(CC)OCCS3)C2)CO1 C#Cc1cc(C(N2CC(C(=O)NOCCOC(C)C)CC2(C)C)=O)ccc1C N1(c2c(S(=O)(=O)NCCC3(C)CC3(Cl)Cl)cncc2)CCOCC(C2CCC2)C1 c1(C(=O)NC2CCCC(NC(C(CC)SC)=O)C2)nc(C)n2ccccc12 c1(OC)cc(C(=O)NC2COCCN(C(c3cnoc3C)=O)C2)c(F)cn1 C1(C(N2CCS(=N)(=O)CC2)=O)(NC(CC(C)(C)C2CC2)=O)CCC(C)(C)C1 c1(C(C2CN(C(C3CC(C(F)(F)F)C3)=O)C2)(F)F)ccc(Br)cc1 CC(C)CC(CCO)NCc1ncccc1C(=O)O c1(C(=O)NC2CCC(N(C(Cc3nc(C)[nH]n3)=O)C)C2)sc(F)cc1C N1(C(C2(CCC)CC2)=O)CCCC2(C1)C(NC(C1CC=CCC1)=O)CCN2C c1(C(C(N2C(C)CC(NC(CCC#C)=O)C2)=O)=O)cc(F)ccc1F c1(C(=O)NC2C(NC(C(CCC)(C)C)=O)C2)c(O)cnc2ccc(OC)cc12 C1(CNC(C2N(C=O)CCC2)=O)CCCC2(CN(C(=O)CSC(F)F)C2)O1 C1(C(=O)NC(C)C(N2CCOCC2)C)CCN(C(C2CC(C)(C)CO2)=O)CC1 C(C)(C)(CC(=O)NC1CCC1CNC(=O)Cc1cnsc1)OC Cn1c(=O)c2c(ncn2CCCC(=O)OC(C)(C)CC(F)F)n(C)c1=O N1(C(c2ccc(C(Cl)Cl)cc2)C(=O)NCC)CCC(C(C)(C)C)CC1C N1(C(CN(C(C2CCN(CCC)CC2)=O)C(C)C)=O)CCN(C)C(CO)C1 N1(C(=O)ON2CC(CC34CCCC3C4)C2)CCC2(CC2)CC1C(N1CCCC1)=O Cc1[nH]nc(C(=O)NC(Cc2ccoc2)C(=O)NC(c2nncn2C)CO)c1C N1(C(c2n[nH]c3c2CSCC3)=O)CCC2CCCCC12 CC(C)C(F)(F)CC(=O)NC1CC(CCNC(c2cnoc2C2CCC2)=O)C1 C1(NC(C2(CC)CCOC2)=O)CCCN(C(=O)CSCC(=O)OC)C1C N1(C(c2cccc(SCC)c2)C(=O)NCCCC2CC2)CCC2(CSC2)C1 CC1CCCc2cc(C(=O)NCc3c(Cl)ccc(Cl)c3Cl)nn21 C1(C(=O)Nc2cccc(NC(CN(C)C3CC3)=O)c2)CCC2C1C2(F)F C(=O)(C1=CCCOC1)N1CCC(NC(c2c(C(C)(C)C)nc(C)s2)=O)C1C CC1=C(C(=O)NC2(C)CCCN(C(C3(C(F)F)CC3)=O)C2)CCO1 C1(NC(CCc2n(C)cnn2)=O)CC2CCC1CN2C(c1[nH]ccc1C1CC1)=O CC1CC(C(=O)NC2(CC(=O)NCc3cnc(O)nc3O)CC2)=NO1 c1(C(=O)NC(C(=O)NC(CO)CCCO)C2(C)CC2)ccc[n+]([O-])c1 C1(C)(C(=O)NCC=CC(C)C)CCN(C(=O)CCn2cnc(=N)[nH]2)C1 N1(C(=O)OC(C)(C)C)CC(O)CC1COC(C1CCCC(O)C1)=O C(C(C(=O)NOCC1CC1)C(C)C)NC(c1c(C)ccnc1)=O C1(C(N2CC(C(C(=O)N(CC#C)CC3CC3)OC)C2)=O)CCC(=O)C1 c1(C(COC(c2c(C(=O)OC)sc(Cl)n2)=O)=O)ccc(O)cc1C C1(CC)CN(C(=O)CC2(C)CC2(Cl)Cl)CCN1C(=O)CC1CCN(C)CC1 c1(C(=O)NCCN(C(c2cscc2SC)=O)CC)cnc(OC)nc1 c1(C(=O)NC(C(=O)NCC(COC)C)CC2CC2)ccc2ccoc2c1 C1(C(=O)NC(CCC=C)(C)C)CCCCC1(C)NC(=O)C(C)[SH2]CC CCCC(C(=O)Nc1ccc(-c2ncc[nH]2)cc1)NC(C)=O C#CCCCC(C)C(=O)NC(CCC)C(=O)N1CC(NC(=O)OC)C1 N1(C(c2cc(CC)n(C)n2)=O)CC(NC(=O)CS(C)(=O)=O)CC(C)C1 N1(C(C=CC(C)NC(=O)Cn2nccn2)=O)CCC2(C=CCO2)CC1 c1(C(N2CC(CCO)(NC(C(C)OC3CCCCC3)=O)C2)=O)cc(=O)n(C)cn1 C(=O)(CCCCc1ccc(F)cc1)N1CCC(NC(C2(CCF)CC2)=O)C1 C#Cc1cccc(C(N2CCC=CC2C(=O)NCC2(CO)CC(C)C2)=O)c1 C1(C(=O)NCCCC(=O)NC(C2CCCCC2)C)CC(C)CC(C)C1 C1(NC(CC2C(C)CCC2)=O)CCC(NC(c2cc(CN(C)C)on2)=O)CC1 C1(C(C)NC(C2(n3cnnn3)CC2)=O)CN(C(=O)COc2ccsc2)CCCO1 CCC(CC(=O)NCC1CC1C(N1CC(C(C)C)C1)=O)CC(C)C C1(C(=O)NCC2N(C(=O)OC(C)(C)C)CC2)CC(F)CN1C(C1CC1C1CC1)=O c1(CCC(N2C3C(NC(CCCCC)=O)C(C3)C2)=O)nc2cccc(C)c2[nH]1 c1(C(N2CC(C)C(CNC(=O)CCCCF)CC2)=O)cc2ccccn2n1 Cc1ccc(=O)n(CC(=O)NCCCCCN(C)C(C23CCC2CC3)=O)n1 N1(C(C(C)n2cncn2)=O)CCC(C2CC2)(NC(=O)CC2(N(C)C)CCCC2)C1 Cc1cc(C)c(C(=O)NCC2CCN(C(=O)CCCN(C)C)C(C)C2)cn1 N1(C(c2c(F)ccc(CC)c2)=O)CCN(C(=O)C(C)SC(F)(F)F)CC(CO)C1 N1(C(CC(=C=C)C)=O)CC2CC(N(C(=O)CSCc3cscn3)C)C1C2 CCCCCC(O)C(=O)N1CCN(C(c2cc(C)c(C)c(F)c2)=O)C(CO)C1 c1(OC)c[nH]nc1C(=O)NC1CCC(N(C(=O)CC2(c3ccccc3)CC2)C)C1 c1(C(=O)OC)cc2cccc(NC3CN(C(=O)OC)CC3(C)C)c2cn1 c1(C(=O)NC2CN(Cc3ncc(OC)nc3)CC2F)n[nH]c2cccc(F)c12 CCCC(C(=O)NCCc1c(Cl)cccc1Cl)S(N)(=O)=O C=Cn1nncc1C(=O)NC1(C)CCN(C(=O)C(C)Oc2ccc(F)nc2)C1 C1(C(N2C(C(=O)NC(C#C)C(C)C)CC(OC)C2)=O)CC12CCOCC2 CC(CS(C)=O)C(=O)NCC1CC(NC(=O)C(Cl)=CCl)C1 Cc1ccc(OS(=O)(=O)Cc2cc(Cl)ccc2Cl)cc1C(=O)N(C)C c1(C(N2CC(SC)C(NC(C3CC4CCC(C3)C4)=O)C2)=O)cc(C)cc(F)c1N c1(CNC(c2csc(C3CCN3CC3CCC(=O)NC3)n2)=O)cc(O)cc(O)c1 C(=O)(CCC(C)(F)F)N1C(C(=O)NCC(C)(C)C2CCCO2)C=CC1 C1(NC(c2ccc(CC)[nH]2)=O)CCN(C(c2ccc(C3CC3)cc2)=O)CC1C C(C(C)C(C)C(=O)N1CC(OCCNC(c2cncc(C)n2)=O)C1)OC C1(OCC)(CN(C(=O)C(=O)N(C)CC2CCCOC2)C)CCS(=O)(=O)CC1 C#CCCCCCCC(=O)NCC1(C)CCN(C(=O)CC2(C)CC2F)CC1 C(=O)(CC(C(F)(F)F)P(C)(C)=O)NCC(COC)NC(c1ccc(C#N)s1)=O C#CC1(NC(=O)CC2CCN2C(=O)C=Cc2ccc(C)cc2)CC2CCCC12 C(CNC(c1c(CNC(C2(n3cccn3)CC2)=O)nnn1C)=O)(CC(C)C)OC C1(CCC)COCCN1C(C1(C2N(C(c3ccccc3CC)=O)CCC2)CC1)=O c1(C(C)C)cnn(CC(=O)NCCOCCNC(C2CCS(=N)N2)=O)c1 c1(C(N2C3CN(C(C4(CC#C)CCOCC4)=O)C(C3)C2)=O)ccc(Cl)c(OC)c1 C1(NC(COCC=C)=O)CCC2(CCN(C(C3CC(C)(C)C(C)(C)C3)=O)CC2)C1 C1(C(=O)NCc2ccc(C(N(CCCCO)C(C)C)=O)o2)NC(=O)OC1C c1(C(N(CCCCN(C(=O)C2=CCCOC2)C)C)=O)ccc(=O)n(CCF)n1 c1(OC)cccc2cc(C(=O)NCC3CCCN3C(C3(O)CCOCC3)=O)oc12 S(=O)(=O)(c1cccc(S(=O)(=O)NC2CCn3cncc3C2)c1)NC1C(C(C)C)C1 C=CC1(C(=O)NCC2(CC)CCOC2)CCN(C(=O)CC(C)C(=O)OC)C1 C12(CNC(C3C(CC)C3)=O)CC(CC)(CN1C(=O)C(C)(C)O)C2 CCC(C(=O)NC(C)(C)C(C)CC(=O)NC(c1cnn(C)c1)CO)C(F)(F)F C(=O)(C(O)CC(C)(C)C)N(C(C)C(=O)NCC(c1ccsc1)C)CCC c1(CC(=O)NCCC(=C)CNC(c2n[nH]cc2C2CCC2)=O)cc(C)ccc1F C(=O)(C(N=[N+]=[N-])C(C)C)NCc1cc(C(=O)NC(C#CCC)(C)C)n[nH]1 C1(C(N2CCN(C(=O)CN(C)C)CC2)C(=O)NC(C)C)CCCC1(C)C C(=O)(CC1=CCN(C)CC1)N1C(C(=O)NC2CCCN(CC)C2)CCCCCC1 C(=O)(C(C)C1OCCc2sccc21)NCC1(F)CC(NC(COC)=O)C1 c1(C(=O)NCC(C)NC(=O)C(F)(F)C2(O)CCC2)cnc2c(c1)CCC(=O)N2 C1(C(N(CCC(=O)NC)C)=O)CN(C(c2cc(C)n(C)c2)=O)CCN1C C(=O)(C(O)CC(C)(C)C)NC(C(N1CC(C)C(C)(CO)C1)=O)C1CC1 C1(C)(COC)CC(c2nnnn2Cc2ccc(F)cc2)(NCC(F)CO)C1 C1(NC(C2CC3(C2)CC3F)=O)CCCC2CN(C(=O)CC3(O)CCCCC3)CC12 c1(C(=O)NC2CC(C)(NC(c3ccc(F)cc3Cl)=O)C2)cc(O)cc(C#N)c1 c1(NC(C23CC2CN(Cc2ncc(Br)cc2Br)C3)=O)cc(F)cc(F)c1[N+](=O)[O-] C1(C(=O)NC(COC)CCO)CN(C(=O)Cc2nonc2C)CC1(C)C N12CC3C=CC1C(C3)OCC2=O.CCC(CC)N(C)C(C1CCCS1)=O c1(C(N2CCC(COC)(NC(C3CCC3)=O)C2)=O)c(C)nn(C)c1C C=CCC(C)(C(=O)N1CCCC1C1(NC(=O)CNC2CC2)CC1)N(C)C NC12CC3CC(CC(NC(=O)CC4CSC4)(C3)C1)C2 c1(OC)nc(N(c2ccoc2C(C)C)CCNC(=O)C2CC2)nc2[nH]cnc12 C1(C(=O)N(c2cnc(Br)cn2)CCO)CSCCN1C(=O)Cc1ccc(Br)cn1 Cc1c(CNC(=O)NCC2CN(Cc3ccco3)C2)ncn1C c1(C(=O)NC2CC3(CCC3)C2O)ccn2nccc2c1 CC12CCC(CNC(NC3CCC4CC4CC3)=O)(C1)OC2.C(C)(C)(C)O c1(OC)nc(C)ccc1C(=O)NCC(C)N(C)C(C1CC1OC(C)(C)C)=O c1(CC)nc(C(=O)NC(c2cn(C)nn2)C(=O)NC(CC)C2CCC2)co1 c1(NC(CCCNC(=O)NC2(C)CCCN2)=O)cc(Cl)ccc1Cl C(CCC(C(=O)NC1CCC1(C)C)NC(C12CSCC1C2)=O)OC O=C(CC1OCc2ncccc21)N(C1CCCCCC1)Cc1cccnc1 C=C=CCCC(=O)NCC(C1CCN(C(=O)C(c2ccc(F)cc2)=O)CC1)(C)O c1(NC2OCCN(C(C(CC(CC)C)C)=O)C2)nc(OC)ccc1[N+](=O)[O-] Cc1cn2cc(C(N3CCN(C(=O)OC(C)(C)C)CC3(C)C)=O)sc2n1 C(=O)(CCC(C)SC)NCC1C(NC(C2CC(OCC)C2)=O)CCC1 CN1CCOCC1C(=O)NCCCC1CCCCN1C(C1SCCS1)=O CC(CC(F)(F)F)N(C(c1cc(C(C)(C)C)n[nH]1)C(=O)NCc1ccco1)C Cc1ccc(C(C)C(=O)N2CC(NC(=O)C(c3cccc(C)c3)F)C2)cc1 N1(CC)CCCC(O)C1C.n1(C2(C(N(c3ccccc3)CC)=O)CC2)cc(C)nn1 N1(C(C(C(C)C)CNC(=O)CCC(F)(F)F)=O)CCCC(C2(C)CC2)C1 C(=O)(C(F)C(F)(F)F)NCCCN1CCN(C(C(CC)n2cccn2)=O)CC1 C1(C(=O)NCC(C(C)(C)C)O)CCN(C(=O)Cn2ncn(C)c2=O)C(C)(C)C1 CC1C(C(=O)NCC(C)(C)CN(C(=O)CC(F)F)C)C1(F)F c1(N2CCC(NCC(C)(Cc3ccccc3)CO)C2)ccc2c(c1)OCO2 N1(C(=O)OCC)CC(C2C(OC)C(C(=O)OC)C2)C2(CC2)C1.C(CC(=O)N)NC N1(c2scc(C)n2)CCN(C(c2ccc(OC)c(OCC(C)C)c2)=O)CC1C C(N=c1nc(N2CC3CC(C)(C)C3C2)c2sccc2[nH]1)C1(C)CC1(F)F C12(NC(c3c(C)nns3)=O)CCN(C(C3(N(C)C)CC3)=O)CCC1C2 N1(C(CC2CC(=C)C2)=O)CCN(C(c2cnc(OC)cc2C)=O)C(C)C1C c1(C(=O)OC)nc[nH]c(=NCC=CCNC(=O)CCC2(C)CC2)c1OC C=CCCCCCCC(=O)NCC(C(C)C(C)C)NC(c1ccc(C(C)=O)o1)=O N1(C(C(C=C)OC)=O)CC2CC(C(=O)NCc3cnc(CC)[nH]3)C(C2)C1 C1(NC(C(C=CCCC)O)=O)CC12CCN(C(c1cc(C3CC3)n(C)n1)=O)CC2 C=CCC(CC(=O)N1CCOCC1CC1CC1)NC(C1CC(C)(C)CO1)=O C1(OC)(COC)CN(C(C2C(c3ccncc3)C2(C)C)=O)C1 c1(C(N(CCn2cc(CCC3CC3)nn2)CC)=O)nc2cnccc2s1 N1(C(CN2CC(C)C2)=O)CCCCC1CCCNC(=O)C=Cc1cc[nH]n1 c1(-c2ccc(C(C)NC3CC(C)N(C(=O)C4=CCCC4)C3)s2)c(F)cccc1F c1(C(N(CC(C)(C)NC(C(C)SC)=O)C)=O)cnc2ccc(F)cc2c1 N1(C(Cc2c(C)cco2)=O)CCCC(C)C1CCNC(c1c(Cl)sc(C)c1C)=O C12(C(=O)NCC3N(C(=O)COC4CCCCC4)CC=C3)CC=CCN1CCC2 CN1CCC(F)(CNC2CCCN(Cc3ccccc3)C2)C1 C1(N(C(c2cn(C3CCOCC3)cn2)=O)CC)CCCN(C(C2(SC)CC2)=O)C1 CC(C)C(C)(CNC(c1ncoc1C1CCC1)=O)NC(C1CCCN1C1CC1)=O c1(OCC)cc(C(N2CCCC2CNC(=O)C=Cc2nccs2)=O)[nH]n1 C#CCC(CC(F)F)C(=O)NCC1CCCN1C(=O)CC1CC(n2cnnc2)C1 c1(C(=O)NC2CC(C(C)(C)C)C2)ccccc1NC(c1nc(NC(C)=O)sc1)=O C1(NC(CCOCC#C)=O)C2CC1N(C(=O)C=Cc1ccc(CC)o1)C2 N1(C(C(N2CCCC(C)C2)=O)=O)CCN(C(=O)C=Cc2cocn2)CC(C)(F)C1 n1(C(C)C)cc(Br)c(C(=O)N(CC(C)NC(=O)C=Cc2cn[nH]c2)C)n1 N1(C(c2nnn(CC)c2C)=O)CCC(NC(=O)CC(C)(O)C2CC2)C(F)C1 c1(C(N2CC(NC(C3CN(CCOC)C(=O)C3)=O)(CO)C2)=O)cncc(Cl)c1C c1(C(N2CCN(C(C(CSC)OC)=O)CC2C2CC2)=O)ccc(Cl)c(N)c1Cl CCC(C)C(O)C(=O)N1CCC(C(C)NC(=O)CN2CCCCS2(=O)=O)CC1 CCC(O)C(C)C(=O)N(CC)CC1CCCN1C(c1cn(CCOCC)nn1)=O Cc1cccc(NC(C2C3CC2N(Cc2cnc(Cl)s2)C3)=O)c1Br CC1(NC(=O)CC(CC2CC2)NC(c2csc(Cl)n2)=O)CCCC1O N1(C(CCS(C)=O)=O)CCN(C(c2ccc(Cn3cccn3)o2)=O)C(C(F)F)C1 S(=O)(=O)(c1ccc(Br)cc1NCc1ncnn1C(C)(C)C)NC(c1ccoc1)C C1(C)(CC(=O)NC2(CN(C)C(C34CCCCC3C4)=O)CC2)CC(F)(F)C1 Cc1cc(C(N2CCOC(C(N3C(CO)CC3CO)=O)CC2)=O)nc(C)c1 CCC(C)(COC)C(=O)NCC12CC(CN1C(=O)CCCOc1ccccc1)C2 C1(NC(N2CCC(C(=O)NCCCC3CCC3)CC2)=O)C2CCC3C(C2)CC13 CCCCC(CNC(C1CC(NC(C)=O)CN1)=O)OC.C(=O)(COC(C)(C)C)N C(=O)(CCC(C)(F)F)N1C(C)(C(=O)NC(CCN(CC)CC)C)CCC1 CC1CC(O)CN(c2cccc(CN3CCOCC3)n2)C1 C1(NC(c2ccc(F)cc2)=O)CCN(C(=O)Cc2csc(Br)c2)C12CC2 CCC(C(=O)N1CCC(NC(=O)CN2CC3CC3C2)C1)C(C)O C=Cn1nccc1C(N1CC(F)CC1C(=O)NC1CC(C(N)=O)C1)=O N1(C(C2(C=C)CCCC2)=O)CC2CC(NC(c3nnc(C)s3)=O)C1C2 c1(C(=O)NC(C(=O)NC(C(C)C)C(=O)N(C)C)C2CCC2)cn(C)ccc1=O c1(C(=O)NCC(C)NC(CCC=C=C)=O)ccc(F)c(S(=O)(=O)NC2CC2)c1 N1(C(c2ccc(CCC)cc2)C(=O)NC2COC2)Cc2ccccc2CCC1C C(=O)(C1=C(C#N)CCC1)NC(C(=O)NCCC(=O)Nc1cn(C)nc1)C1CC1 CC#CC1CCN(C(C2CN(C(C3(N(C)C)CC3)=O)CCO2)=O)CC1 N1(C(c2n(C(C)C)ccn2)=O)CCCC2(C1)CN(C(=O)CCN1CCC(F)C1)C2 c1(C(=O)NCCN(C(C(C(COC)C)C)=O)C(C)C)cnc2c(c1)CCC(=O)N2 CCC(CC(F)(F)F)C(=O)NCCCC(C)NC(c1nc(C2CC2)cs1)=O c1(C(C)C)ccc(Cl)cc1C(=O)NC1CC2CC(NC(=O)CCC(C)C#N)C2C1 C(CCC(=O)NCC1(C(=O)NCCCn2ccnn2)CC1)OC Cc1[nH]c(=NCc2c(Cl)cnn2C)sc1S(=O)(=O)N1CCC2(CC2)C1 N1(C(c2cc(C(=O)OC)n(C)c2)=O)CCN(C(=O)C(O)CSC)C(C2CC2)C1 N1(C2CCC(NC(COCCCOC)=O)C2)CCN(C(=O)CCOC)CC1 c1(C(=O)NCc2cccnc2)ccc2c(c1)CCCN2C(C1(NC(C)=O)CC1)=O C1(C(=O)NCC2(CC)CCCO2)CN(C(=O)C(OC)OC)CC12CC2 C#Cc1ccc(C(N2CCC2CC(=O)NCc2ncnn2C2CC2)=O)cc1 c1(NC(C2N(C(C(CC)O)=O)CC(C)C2)=O)cc(F)c(F)cc1I C=CCC(C)(C)CC(=O)N1CC(N=[N+]=[N-])CC1C(=O)NC(C)C(C)F c1(C(=O)NC(C2CCOC2)CNC(CCC(=O)N(C)C)=O)ncc2[nH]ncc2n1 C=CC(C)(C)CC(=O)N1CC2(CC2)CC1CNC(C1CCC(F)(F)CO1)=O C(=O)(CC1OCc2ccccc21)NCCN(C(CCn1c(C)csc1=O)=O)C C1(CNC(C(CCC)NC(N)=O)=O)(CO)CCCN(C(C2COCCN2C)=O)C1 N1(C(C(CCC)C)=O)CC2CCC(C1)N(C(=O)C(c1ccccc1Cl)O)C2 O=C1NC(Cc2cccc(F)c2)C(=O)N1c1ccc(O)cc1Br N1(CC(N2CCC(CNC(c3cn(C(C)C)nc3)=O)C2)=O)C(=O)CSC1=S CCCCC(CC)CC(=O)NC(CCN(C(=O)Cc1ncnn1C)C)C(C)(C)C C1(CNC(CC=C)=O)CCC2(CCC2)C1NC(=O)CN1CCOCC1 Cc1ccc(C#N)c(N2CCN(C(=O)C(C)(C)c3ccccc3)CC(O)C2)n1 N1(C(C(CCSC)O)=O)CC2CCC1C1CN(C(c3ccc(Cl)o3)=O)CC21 c1(NC(C2CC(NCc3c(Br)cc(F)c(F)c3F)C2)=O)ncnc2[nH]c(Br)nc12 C1(NC(CC(C)C(F)F)=O)CCC2CCN(C(c3ncn4c3CCC4)=O)C12 N1(C(C(C)OCCCC)=O)CCC(NC(=O)CC2CC(=O)NC(=O)C2)C(C)C1 Cc1cc(F)cc2[nH]c(C(N3CCC3CNc3ncnc4c3COC4)=O)cc12 CCC(C)(CNC(=O)CCN1CCCC1=O)C(=O)Nc1cc(OC)ccc1C N1(C(CCCNC(C)=O)=O)Cc2n[nH]cc2C1C(=O)NCC(C)F CCCC(C)(CC)C(=O)NCCC(C)CCNC(=O)C(C)NC(n1cnnn1)=O CC1CN(C(C2CC(N3CCOCC3)C2)=O)CC1NC(C1CN(C2COC2)C1)=O C1(C(N2CCC(C(CC)CC)C2)=O)CCCCN1C(C1C2CCC(F)C12)=O N1(C(c2c(CC)occ2)=O)CCC(O)(CNC(c2cnnc(N(C)C)c2)=O)CC1 CC(C)(C)CCCCCC(=O)NCC1CC(NC(=O)CNC(N)=O)C1(C)C N1(CC(C2CCC(C)O2)=O)CCCN(C(c2ccc3c(c2)COC3)=O)C(C)C1 c1(C(N2C(C(C)NC(c3ncoc3C3CC3)=O)CCC2)=O)ccc2c[nH]nc2c1 C(CCC(O)C(=O)N(C)CCC1CCCO1)NC(CCC=C(C)C)=O N1(C(=O)C(F)C2CCOC2)CCN(C(=O)CCc2ccsc2)CC2(CC2)C1 Cc1ccc(NC(=O)C(=O)NCCSCS(C)(=O)=O)cc1C(F)(F)F.C1CO1 N1(C(C(C2CC2)OCC)=O)CC(OC)C(NC(=O)C(c2ccccc2C)(F)F)C1 C(CC(=O)N1CC(C)(C)CC1CO)(C(F)(F)F)NC(C1C(=C)C1)=O C1(NC(=O)Cn2cc(CO)nn2)COCCN(C(c2cnc(S)n2C2CC2)=O)C1 C12(CNC(c3cc(CCC)nn3C)=O)CCCC1CN(C(=O)CSC)C2 c1(C(=O)NC(C)(CNC(=O)CC2(C(F)F)CC2)C2CC2)ncnc2ccsc12 CC1(O)CON(C(=O)C2CCCCN(C(c3nccc4cc[nH]c34)=O)C2)C1 Cc1cnnc(O)c1C(=O)NC1COC2(CNC(C3(C#N)CC3)=O)CC1C2 c1(NC2(c3c(C)cccc3C)CC2)ccc(Cl)nc1OC.C=C1CC2N(C1)C2=O N1(C(c2c(CC)cnn2C)C(=O)NC(C)(C)CC)CCNC(=O)CC1 c1(C(=O)NCC23CC(CN2C(c2cc[nH]c2)=O)C3)ccc2c(c1)NC(=O)CC2 N1(CCCCCNC(C(CC)N(CC)CC)=O)CCN(C(=O)CC(C)(F)F)CC1 Cc1nc2ncnn2cc1C(=O)NC1(CNC(C2CCOC2)=O)CCCCCC1 CCCC(C(=O)NC1(n2cccn2)CCN(C(C2(C(N)=O)CC2)=O)C1)S(N)(=O)=O n1(C(c2ccncc2)C)nc(-c2ccccc2Br)nc1-c1cc[nH]n1 N1(C(c2c(CCC)nco2)=O)CCC2(CC1)CCN(C(=O)C(C)(O)C1CCC1)C2 c1(NC(=O)NC(C)C(=O)N(CCCCNC(c2cnoc2)=O)C)ccc(Cl)cc1 Cc1cc(-c2cn(C3CCN(C(C4CCS(=O)(=O)N4)=O)CC3)nn2)ccc1Br CC1CC(Nc2cc(COc3ccccc3)ncn2)C(C)O1 C#CCC(C)(CC)C(=O)N(C)CCOCCC(=O)N1CC(c2nocc2C)C1 N1(C(COCCC)=O)CC(CNC(c2cccc(-n3cc(C)cn3)c2)=O)C(C)C1 N1(C(CC=C=C)=O)CCCC(C(=O)NCC(C)CCO)C1CC N1(C(c2c(OC)nn(C)c2)=O)CC(N(C)C(C2C(Cl)(Cl)C23CC3)=O)C2(CC2)C1 N1(C(=O)NC)CCC(C(N2CCC(CNC(C3CC(C)(F)C3)=O)C2)=O)C1 c1(C(N2CCC(C3C(C)(C)C3)C2)=O)cc2ccoc2cc1F c1(C(N(C2CCN(C(c3nnsc3C)=O)C2)CC#C)=O)noc(CC)c1C Cc1cnc(C(=O)NC(C2CC2C(=O)N(C(C)CO)CCN(C)C)C)cn1 c1(SC)ccc(C)c(C(=O)N(C2CCN(C(=O)CCS(C)=O)CC2)CC2CC2)c1 c1(NC(CC(CC)N(C(=O)CN(C2CCCC2)C)C)=O)cccn2nccc12 c1(C(C)NC(Cn2cc(CNC(C3(C)CC(=C)C3)=O)nn2)=O)nccc(C)n1 c1(C(=O)NC2C(NC(C3(C)CCC3)=O)C2)ccncc1I C(=O)(C1=Cc2ccccc2C1)NC1C(CNC(=O)CCCc2ncco2)CCC1 N1(S(c2c(C)onc2)(=O)=O)CCC2C(CCN2C(c2c(F)cc(Cl)cc2F)=O)C1 c1(C(N2C(CC(=O)NCC(C(=O)OC)(C)O)CC(F)C2)=O)ncc2ccccn12 C(=O)(C(CC)C(C)C)N1CCC(C(=O)NCCCC)(CC)C1 C1(C(N2CCCC(CCC(=O)NC3C(C)CCC3C)C2)=O)CC2(CCC2O)C1 N1(C(C(C=C)O)=O)CC(NC(=O)COCc2ccnn2C)CC12CCC2 N1(C2(C(N)=O)CC2)CCN(C(C2CC=CC(O)C2)=O)CC1=O Cc1cccc(-n2ncc(C(=O)NCC3CC3NC(=O)CC3CC=CC3)c2C)c1 N1(C(C(n2ncc(C)c2)C)=O)CC2CCCC(N(C(=O)CC(F)(F)F)C)C2C1 N1(C(c2cnc(C)s2)=O)CCC2CCN(C(=O)C=CSCc3ccco3)C2C1 N1(C(C2=NNC(=O)C2)=O)CC2CC1CCC2NC(=O)CC1CCC(F)(F)C1 C1(C(=O)NCC(c2cccc(C)c2)=O)Cc2cn(C)nc2C(C)C1 CCC(CC(=O)N(CCNC(=O)Cc1cnn(C)c1)C(C)C)NC(=O)OC(C)(C)C CCC(C)(C)CC(=O)N1CCC(C)(CNC(c2nccc(C)c2F)=O)CC1 N1(C(C(C)C2CCC2)=O)CC2CCN(C(c3csc4ccccc34)=O)C2C1 C(=O)(C(CCSC)NC(=O)CC(C)n1ccnc1)N(CC(C(=O)OC)C)C C1(NC(CCNC(C)=O)=O)CC2CCC(C1F)N2C(=O)CCOC(C)=O N1(CC(=O)NCC2C3N(c4c(OC)c(C)ncn4)C(CC3)C2)CCCCCCC1=O C(=O)(CS(=O)(=O)CC(C)C)NCC(CN(C(C=C(C)c1ccccc1C)=O)C)O N1(Cc2c(OC)nccc2)CCC2CN(C(c3occc3Br)=O)CC2C1 N#CC1(NC(c2cccnc2S)=O)CCN(C(=O)Cn2ccnc2)C1 N1(C(C(C(C=C)C)C)=O)CCOC2(C1)CN(C(=O)CC1(C3CC3)CC1)C2 C1(CNC(C2C(C(=O)NC3CC(C(=O)OC)C3)C2(C)C)=O)CC12CC2(F)F C1(c2cn(C3CC(C(=O)NC4CCCCO4)C3)nn2)(OC)CCOC1.c1cccnc1 c1(C(=O)NC2CC(O)(CNC(CCC3N(C)CCC3)=O)C2)nccc(Cl)c1F NS(=O)(=O)c1ccc(C(N2CCN(C(=O)C=CI)C(CCO)C2)=O)o1 C#Cc1cccc(C(=O)N(C(C)(C)CC(=O)NCCn2cccnc2=O)C)c1 C(CCCC(C)NC(=O)CNC(N)=O)NC(C(C)OCc1ccccc1)=O CC(=NOCC#N)C(=O)NCCN(C(=O)COCC1CCCC1)C c1(C(N(C(CC)CC(=O)N(C)C)C2CC2)=O)cccc2c1OCCN2 C1(n2cc(CNC(c3ccccc3Cl)CO)nn2)CCCCCC1O C1(CC=C)(NC(C2CCOC2)=O)CN(C(=O)COC2CCOCC2)C1 C1(NC(c2ncn(C(C)C)n2)=O)C=CCN(C(C2(c3cccc(Cl)n3)CC2)=O)C1 C1(NC(C=CCOC)=O)CCC12CCN(C(c1cccc(C3CC3)c1)=O)CC2 C1(NC(C(CNC(C)=O)(C)C)=O)CCCN(C(=O)CCc2nncn2C)C1C C(=O)(CCS(C)(=O)=O)N(C)CC1CN(C(=O)Cc2ccccc2F)CCO1 c1(CC=C)ccccc1C(N1CCOC(CC(=O)N(CC(=O)OC)CC(C)O)C1)=O N1(C(CNC(CCC)=O)=O)CC2(COC(CNC(C3(OC)CCCCC3)=O)C2)C1 C1(CC(N2C(CCNC(CC3(OCC)CCC3)=O)CCC2)=O)CCCOCC1 C(=O)(C1CC(=O)c2ccccc21)N(C)CC1N(C(C(C=C)OC)=O)CCC1 c1(NC(C2C(C(=O)Nc3cc(O)cc(Cl)c3)C2)=O)ccc2oc(O)nc2c1 N1(CCOC)CCn2ncc(CNS(C)(=O)=O)c2C1.n1(CC=O)nc(C)cc1C CC1CC(C(=O)NCC2(O)CC(CO)C2)N1C(=O)CC1CCOC1=O c1(C(N2CCC(NC(CC(CCC)C)=O)(CO)C2)=O)ncc([N+](=O)[O-])cc1C c1(C(C)N(C)C(c2coc(CNC(=O)C(C)(C)C3CCOC3)n2)=O)cnnn1C c1(CC(=O)NC2CN(C(C3C(OC)CCCC3)=O)CC2C)ccc2c(c1)CCO2 C(=O)(C1=CCS(=O)(=O)C1)NCC(CC(C)C)(C)NC(C1CCC(C)(C)O1)=O CCC(CC(=O)NC(CNC(=O)C(C)C(C)O)C(C)(C)C)C(C)C c1(C(=O)NC2C3(CN(C(C(N4CCNC4=O)C)=O)C3)CC2)cnc2ncccn12 c1(OC)ccc(COC(C2(C)CCCS2(=O)=O)=O)c(F)n1 Cc1ccncc1C(N1CCC(O)C1C(=O)NCC(=O)N(C)C)=O N1(C(c2cncc(OC)c2)=O)CCN(C(C2CC(C)(C(C)(C)C)C2)=O)CC1CO c1(CN(C(CCC)CO)C=O)c(Cl)cnn1C C(c1cccc(F)c1Cl)=CC(N1CC(NC(C(C)=CC)=O)CC1(C)C)=O C1(C(=O)NC(C(C)C)C2CC2)CC1C1CN(C(=O)CC2CCCOC2)C1 c1(C(=O)OC)cc(C(N2CCC(CNC(=O)CC3C=NN(C)C3=O)C2)=O)oc1C C(c1cncc(C)c1)=CC(=O)N(C(CC)CNC(=O)C(C)Oc1cccnc1)C C(=O)(CCCCC(F)F)NCC1C=CC(NC(c2cc(OC)n[nH]2)=O)C1 c1(CC(=O)OC(C2CC2C(c2ccccc2)NC(CCC)=O)=O)cnc(C)s1 c1(C(=O)OCC)cc(C)nc(N2CCCC(CO)(NC(=O)C(C)=C(C)C)C2)n1 c1(NCC2CC(=C)C2)[nH]c(=NC(CCO)C2CCC2)nc2ncn(CC)c12 N1(C(Cc2nc(C(C)C)sc2)=O)CCN(C(=O)C(C(C)C)NC(N)=O)C(CF)C1 c1(C(N(C2CC(NC(c3cc(OC)n[nH]3)=O)C2)C)=O)cccc2ncc(C)n12 Cc1cc(C(N2CCCCC2c2cccnc2)=O)c(N)c(F)c1 Cc1cc(F)cc(C(=O)NCC2CC(NC(C3(C)CCCC3(F)F)=O)C2)c1O N(C1CCOc2ccc(Br)cc21)C(c1nccc(Br)c1F)=O N1(C(C(C)NS(CC)(=O)=O)=O)CCCC2CN(C(c3cn(C)c(O)n3)=O)CC12 c1(C(N(CC(C)C#N)C2CC2)=O)c[nH]nc1CCNC(=O)C=Cc1cocn1 c1(NC(C2N(C(c3scc(OC)c3)=O)CC2)=O)cc(C(F)(F)F)c(Cl)cc1Br c1(C(N2CCC(C3N(c4snc(C)n4)CCCC3)C2)=O)ccc(C)c(F)c1 C1(NC(N2CCC(O)(C(C)CN(C)C)C2)=O)CC(=O)NN(C(=O)OC(C)(C)C)C1 C(C)(C(C)n1cncn1)NC(CN(CCOC)C(C1C=CCS1)=O)=O CC(C)(CNS(=O)(=O)CC1CC2OCCC2O1)CCC#N c1(N2CC=CC(NC(C(CC)n3ccnc3)=O)C2)ncc(Br)c(O)n1 CCCCC(C(=O)NC1CCC(NC(=O)C(N)=O)CC1)ON=C(C)C Cn1[nH]c(=NC(=O)NCC2(COc3ccc(Br)cc3)CCCC2)cc1Br c1(OC)ccc(O)cc1NC(C1(NC(=O)Cc2cc(C)n(C)n2)CSC1)=O Cc1nnc(CC(=O)NC2(C)CC(NC(C3(F)CCOC3)=O)C2)o1 c1(NC2CCN(C(c3c(OC)ncc(F)c3)=O)CC2F)ncnc2[nH]ccc12 n1(CCC)cc(CNC(C2OCCC2NC(c2ccc(Cl)o2)=O)=O)nn1 C1(NC(c2nccc(C)c2)=O)CC(F)CN(C(=O)CC2C=NN(C)C2=O)C1 c1(C(C(=O)NCCOC)N(c2cccs2)C)ccc(OCC)cc1.CCC(C)(C)O CCCC(C(=O)OC)C(=O)NC1C2CN(C(c3cnn(C(C)(C)C)c3)=O)CC12 N1(C(C2(OC)CCN(C(C(CCCC)CC)=O)C2)=O)CC2(COC(C)(C)C2)C1 c1(C(=O)NCC(CC=C)NC(c2cscc2Cl)=O)cncnc1C C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)NCC1CN(C(c2c(CC)cc[nH]2)=O)C1 c1(CC)cc(C(=O)N(CCN(C(=O)CC(O)CN(C)C)C)C(C)C)n(C)n1 Cc1cc(C(N2CC3C(CNC(=O)Cn4cccn4)C3C2)=O)ccc1Br Cc1nc(-n2cccc2)sc1C(=O)NC1CCC1CNC(c1cnc(S)nc1)=O C(C(CC)(CC)NC(=O)COc1cccc(O)c1)NC(C(CC)N(C)C)=O c1(OC)ccc(Cl)cc1-c1ccc(COc2cc(C)cnc2OC(C)C)cc1 c1(C(=O)NCC2OCCN(C(CCC(=C)Cl)=O)C2)cc([N+](=O)[O-])c(C)cc1C N1(CC(F)(F)F)CC2(CCC(Cc3nn[nH]n3)CC2)C1.c12nc-1no2 C12(C(N3CCC(F)(CNC(c4ccc(C)cc4)=O)C3)=O)CCCC1CCC2 N1(CCNC(CCCNC(C(C)Cn2cccn2)=O)=O)CCC(C)(C)C1 C1(CNC(C(CCC)(C)O)=O)CN(c2ncccc2C(=O)OC)CCC1(F)F N1(C(CCC2(C)CC2)=O)C(CNC(C2CNC(=O)O2)=O)CC2CCCC12 n1(COC)nccc1C(N1CC(N(C(=O)Cc2ncc(C)s2)C)C1)=O NS(=O)(=O)c1cc(C(=O)NCCNC(c2ccc(-n3cccc3)cc2)=O)c(Cl)o1 C1(C)(CC)C=C(C(=O)NC2CCCCCC2C(=O)NCc2cnccc2Cl)C1 CCC(CC)C(C)C(=O)NCC1CCCC1NC(C12CC=CCN1CCC2)=O N1(CCN(c2nc(C)sc2)C)CCN(S(=O)(=O)C2CC2)CC1 c1(CC(=O)NCC(CC)NC(=O)C=Cc2cn(C)nn2)oc2ccccc2c1C c1(C(C(N2CCC(Cn3cc(CCN(CC)CC)nn3)C2)=O)C)cncc(F)c1 N1(C(c2noc(CC)c2C)=O)CCC(C)(NC(c2cc(CC)no2)=O)CC1 C1(C(N(C(CCO)C(F)F)C)=O)CN(C(c2ccc(F)cc2F)=O)CC1C1CC1 c1(C(=O)NC(CNC(C(CC)C)=O)C(C)(C)C)cccc2occc12 c1(OC)ncnc(C)c1C(=O)NC1CCC(N(C(=O)COC(C)C)C)C1 C1(CC)CC2CC(OC)C2C1.N12CCC(CC1)C(C)C2=O.c12cccc(c1)C2 c1(C(N2CCC(NC(C3CC4(CC(C)(C)C4)C3)=O)C2)=O)cc2c(=O)[nH]ccn2c1 c1(C(N2CC(N(C(c3c(OC)nccc3)=O)C)C2)=O)cc(C)c(Cl)cc1Cl C(=O)(C(C)C(=O)N(C)CC1(O)CN(C(=O)C(C)Cc2cnco2)C1)OC c1(C(N2CCC(NC(=O)CCF)C(O)C2)=O)nc(Br)n2c1COCC2 CCC(CC)(CC)C(=O)N1CC(Nc2nc(C)ncc2C)CC(C)(C)C1 CC1(F)CN(C(c2csc(S(N)(=O)=O)c2)=O)CCN(C(C2CC=CC2)=O)C1 c1(OC)cccnc1CNC(=O)C(O)CNC(c1cnsc1)=O C(=O)(CCC(C(=O)N1CC(CN)CC12CCC2)C(C)C)OC c1(C(=O)OCC)cc(Br)ccc1NC(C1CCCN1Cc1cncc(Br)c1)=O C1(CNC(C(N2CCOCC2)C)=O)CC(NC(c2cc(C(F)F)cs2)=O)C(O)C1 C1(C(=O)NCC(COC)O)CC12CCN(C(C1CC(SC)C1)=O)C2 C#CCC(CC(F)F)C(=O)NC1CN(C(c2cc(C)c(C)o2)=O)C(C)(C)C1 N1(C(C(CCSC)O)=O)CCOCCC1C(N1CCCCC1CO)=O C1(NC(CCN(C)CCO)=O)CCC(NC(=O)C(C)(C)C2CC2)CC1 c1(C(N(C(CN(C(c2c(CC)non2)=O)C)C)C)=O)cnc2c(c1)CCCC2 C12(CNC(C=Cc3n(C)cnc3)=O)CCCC1CCN2C(=O)C=Cc1nccs1 C=C=CCC(=O)N(C(c1ccccc1)CNC(C1(F)CCCC1)=O)C N1(C(c2c(CC)occ2)=O)C2CC=C(C(=O)N3Cc4cccc(O)c4C3)C1CC2 S(=O)(=O)(CC(=O)N1CCC1CC(=O)NCC1(C2CC2)CCCO1)NCC c1(C(N(CCC(C(C)C)NC(=O)CNC(N)=O)C)=O)cncc2c[nH]nc12 Cc1c(C(N2CCC(N(C)C(C3CN4CCCC3C4)=O)C2)=O)cncc1F c1(OC)cc(CNC(=O)CCN(CCO)C(c2cc(O)cs2)=O)ccn1 N1(C(c2n[nH]c(C)c2C)=O)CCC(NC(=O)CC2CCCNC(=O)C2)C(C)(C)C1 c1(NCCN(C(C2C(C)CC=CC2)C(=O)NCC(F)F)C)cc2ccccc2o1 C(=O)(C=CS(C)=O)NCCC1(CNC(C(C)Cc2ccco2)=O)CC1 N1(C(c2c(C)ncn2C)=O)CCC(C2CC2NC(=O)C(C)c2cc[nH]n2)CC1 N#CCCCC(=O)NCCCN(CCO)C(C1CCCCC1c1nc(S)n[nH]1)=O C(=O)(C1CCCn2nccc21)NC1C2(CC(NC(c3ccnnc3O)=O)C2)C1 Cc1[nH]nc(C(=O)NCC2CCCN2C(c2cnnn2C)=O)c1C(F)(F)F c1(OCC)ncnc(N2CC3CC2CN3C(c2cc(C)cc(C)c2)=O)c1C c1(NC(=O)NC(c2ncc(Cl)n2C)C)ccc(N)cc1-c1ccccc1 C1(C(N(CCN(C(CCCC(=O)NCC)=O)C)C)=O)Cc2cc(C)ccc2S1 c1(C(C2CCN(C(C(=O)Cc3cccs3)=O)CC2)O)ccc(O)cc1 c1(C(C)C)ccc(NC(c2c(NC(=O)CCCCCl)cccc2F)=O)c(C#N)c1 C1(C)(C(=O)NCCOCCN(CCCc2cccc(OC)c2)C)CCC(C)=C(C)C1 c1(C(=O)NCC2N(C(c3ccc(C)nn3)=O)C3CCC2C3)c[nH]c2ncccc12 C1(C(N(CC(C(=O)OC)C)C)=O)CCOCC1NC(=O)Cc1cnoc1 CCC(CCC(=O)N(C)Cc1ccc(F)cc1)NC(=O)C(C)C#N C1(C(C)C)CN(C(=O)CC2CCC3CC3C2)CCN1C(c1[nH]ccc1C1CC1)=O c1(NCC(CO)OC)ncccc1S(=O)(=O)NCC1CCCCS1(=O)=O C(=O)(CC(C(F)F)c1ccccc1)NCC(CC)NC(c1oc(Br)nc1C)=O C1(CCNC(c2c(C)con2)=O)CSCCN1C(=O)C(N1CCC(O)CC1)C c1(C(=O)NC2C(C)CN(C(c3cnc(S)[nH]3)=O)C2)cc2cncn2c(O)n1 N1(C(c2cncc(OC)c2)=O)CCC(CNC(=O)COC2(C)CCC2)C(C)C1 CC(CNC(C1CC(N(C)C)C1)=O)C(=O)N1CCC(OCC(=O)NN(C)C)C1 c1(C(=O)NCC(CCCC)NC(=O)CCc2nc[nH]n2)cc2nc(=O)ccn2[nH]1 C12(NC(=O)CN(C(=O)Cc3ccnc(O)c3)C3CC3)CCCN(CC1)C2 c1(C(COC)NC(C2CC2c2cccnc2)=O)ccc(OC(F)F)cc1 c1(NS(C)(=O)=O)ccc(CNC(c2nc(C)sc2C)=O)cc1.C12(F)CN(C1)C2 C1(C(N(CCOC)CCNC(=O)Cc2nocc2C)=O)CCC(C)(C)OC1 c1(C(=O)NCCN(C(CC(C)C2CCCO2)=O)C)ccc2c(=O)ccoc2c1 C1(C(=O)N)CC2CCC(C1)C2(F)F.C1(CSCC(=O)NC2(C)CC2)CCCO1 C1(CNC(C2CC(=C)C2)=O)CC2CCCC(C1)N2C(=O)C=Cc1ccc(CC)o1 c1(C(N(C(C)C(=O)N(C)CC2CCN(C)C2)CCC)=O)ccn2nccc2c1 N1(C(c2cc(Br)cs2)=O)CCC2C1CCN2C(c1cncc2c1CCC2)=O N1(C(C(CC(C)C)F)=O)CCC2CCCC(C1)N2C(c1cc(F)c(O)c(F)c1)=O Cc1cc(C(=O)NCC2(F)CN(C(=O)CNC(=O)OC(C)(C)C)C2)oc1Br N1(C(C(CC)(C)CC)=O)CCC2(CC1)CC(C)N(C(C1CC(OC)C1)=O)C2 C1(CC(=O)NC2(C(=O)OC)CCC2)C(NC(c2nncn2C(C)C)=O)CC1O C1(NC(c2nc(C(C)C)sc2)=O)CN(C(=O)C(C)(C)c2ccnn2C)CC1F O=C1CCCc2sc(N(C3CCCCC3)C(c3ccc(O)cc3O)=O)nc21 N1(C(C(CC)COC)=O)CCC(C(=O)NCCCOCCOCCO)C(C)C1 C1(C(=O)NCC2(F)CCC(NC(c3ccc(OC)cn3)=O)C2)CC2(C1)CC2(F)F C(=O)(CC(O)C(C)CC)NCC(CCNC(CC1(OCC)CCC1)=O)OC CC(C(=O)NC1CC2(C1)CC2NC(=O)CSCC(F)(F)F)S(C)(=O)=O C(=O)(CCCC(C)CC)NC1C2CN(C(C3N(CCCC)CCCC3)=O)C1C2 c1(C2(NC(C3C(C(N4CCOCC4C4CC4)=O)CC3)=O)CC2)ccc(F)cc1Cl CCC(C(=O)NCC#CCNC(C1(C(F)F)CCCC1)=O)C(C)(C)CC C1(F)(C(N2CC(CNC(CCOC)=O)C(C)(C)CC2)=O)CS(=O)(=O)CC12COC2 C1(NC(C=CCC)=O)CN(C(c2sc(C)nc2C)=O)C(CC)(CC)C1 c1(CNC(=O)NC(C2(C(=O)OCC)CCCC2)C)c(C)nn(CC)c1OCC C(CCC(C)(C)COC(=O)CC1OCCOC1(C)C)OC c1(C(C)C)nc2[nH]ccc2c(=NCC(C)(C)C2CCCO2)[nH]1 c1(C(C(=O)N(CCCO)C(=O)OC(C)(C)C)(F)F)ccc(C(F)(F)F)cn1.CCO C1(C(=O)NC2C(NC(c3nccc(Br)c3O)=O)COC2)CCn2nccc2C1 CCC(c1cccc(Cl)c1)=CC(=O)N(C)CCNC(=O)C(c1cccc(F)c1)O CC1(C(=O)NCc2ccc(-c3ccncc3)cc2)CCC(N)C1 C1(CNC(CC2C(C)(C)COC2)=O)CN(C(C2(C(F)F)CC(O)C2)=O)CC1(C)C c1(CC)c(C(N2CCCCC(NC(C3CNC(=O)N3)=O)C2)=O)oc2ccccc12 C(=O)(CCCS(C)(=O)=O)NCC1(NC(=O)Cc2ccno2)C(C)CCCC1 c1(C(N(CCCCN(C(=O)C(F)C2CCOC2)C)C)=O)c(C(F)F)cnn1C CC1CCN(C(c2cc(O)ccc2F)=O)CC1CC(=O)N(C1(CCO)CC1)C C#CC1CN(C(C2CC(=O)CS2)=O)CCN1C(C1CC(=C2CCC2)C1)=O C1(C2CCCO2)(C(N2CCC(CNC(c3nc(Cl)c(Cl)s3)=O)C2)=O)CCOCC1 C1(N(C)C)CC(C(=O)NC2CC2CNC(=O)Cc2cnc[nH]2)C1 S(=O)(=O)(c1ccc(F)c(Cl)c1)NCC(=O)NCCCC(=O)NCc1ccccc1 C1(C(=O)NC(C)(C)C)CCN(C(c2ccc(CO)o2)=O)CCO1 C1(N(C)C(c2ccoc2)=O)CC2CC1N(C(c1cn(C3CC3)cn1)=O)C2 c1(C(C(=O)NC(CNC(c2cnc(C(C)C)s2)=O)C2CC2)(F)F)ccccc1F CC1CN(CCNC(=O)C(=O)NC2CC2(c2ccccc2)C)CC1CN C1(C(C)NC(CC(=O)NCC)=O)CN(C(c2ccncc2F)=O)CCO1 CC1CN(C(=O)CCc2cnco2)CC(C)C1NC(c1c[nH]nc1C1CC1)=O C1(CCOC)(NC(c2ncc(C)cn2)=O)CCN(C(C2CCOC(C)C2)=O)CC1 C(=O)(C(CC)C(=O)N1CC2(C)CC1(C(=O)NC1CN(C)CCC1O)C2)OCC c1(C(N2CCN(C(CNc3cccc(C)n3)C)CC2)=O)ccc2[nH]ccc2c1 C1(C(N2C(CNC(=O)C3=CCCC3)CC3(CCC3)C2)=O)CCc2ncccc2C1 c1(OC)ccc(F)c(-c2cnc(Oc3ccc(C)nc3F)nc2)n1 CC1CN(C(c2ccc(C(F)F)cn2)=O)CC(C)C1NC(C1(C#N)CC1)=O N1(C(c2cc(COC)[nH]n2)=O)CCCN(C(C2CCCN2C=O)=O)C(C(C)C)C1 c1(CNC(=O)Nc2c(C(=O)OC)nn(C)c2)c(C(F)F)nn(C)c1Cl CC1CN(C(c2cscc2F)=O)CCC1NCCOCC1CC1 N(C1c2cc(C)ccc2CC1C)C(c1c(CC)nn(C)c1)=O CN1CCN(C(c2ccc(C#N)o2)=O)CC1C(=O)Nc1cccc(CCO)c1 c1(C(N(CCCNC(c2cccn2C2CC2)=O)CC)=O)c(C)[nH][nH]c1=N c1(C(N2C(C)(C)CC(CNC(=O)CCNC(N)=O)C2)=O)ccc2c(c1)C=CCC2 C1(C(=O)NCCN(C(=O)C2=CS(=O)CCC2)CCOC)CCc2ncc(C)n2C1 N1(C(C(CC)(C)O)=O)CC(F)(F)CC1C(N1CCC(C(C)(C)C)CC1)=O N1(C(C2(C)C(C)CCC2)=O)CCCC(C2CN(c3ccn4c(Br)cnc4n3)C2)C1 c1(OC)[nH]c(=N)nc2sc(C(=O)NCC3CCCN(C(C4CCOC4)=O)C3)cc12 c1(C(=O)NC(C(C(C)C)NC(C2CC3(CC(=C)C3)C2)=O)C)cccc2ccsc12 NS(=O)(=O)c1ccc(NC(C2COCCN2C(c2cc(Br)ccc2F)=O)=O)cc1 C(C(=O)NN1CCC(C(F)(F)F)CC1)=Cc1cc(C)c(Br)cc1 c1(OC)cc(C(=O)NCc2cc[nH]n2)c(NCc2cc(SC)ccc2O)cn1 c1(C(=O)NC2CC(CNC(C3C(C(C)C)(CC)C3)=O)C2)cc(F)cc(C)c1N c1(C(=O)NC2CCC(N(C(C=COCC)=O)C)C2)cc(C)nc(C)n1 C1(C(N2CC(C)NC(=O)C2)=O)CCCN2CCCCC12 C1(NC(C2=CCN(C(C(C)(C)OC(C)=O)=O)C2)=O)CCn2ccnc2C1 C1(C(=O)NCCN(C(c2cnn[nH]2)=O)CC)(C(=O)NC2CC2)CCOCC1 C12CCCN(C1)C(=O)OCCOC2.c1(OC(=O)CO)ccc(Br)s1 CCCCCC(C)C(=O)NC1CCN(C(c2n[nH]c3c2CCCC3)=O)C1 c1(N2CCC(CC(C)(C)C)C2)nc(N2CCCC(C)(C)CC2)nc2c1SCC2 C(=O)(C#CC1CCCC1)NCC(CC)(C)C(=O)NC(C)Cc1cn[nH]c1 C1(C)(C(=O)NCc2ccc(C(NOCC=C)=O)cn2)CCC(=O)CC1 C(=O)(C1CCCc2ccnn21)N1CCC2(CCN(C(=O)C=CC(F)(F)F)C2)C1 N1(C(C2(N(C(Cc3cc(C)n(C)n3)=O)C3CC3)CCC2)=O)CC(C)C(C)C1C c1(SCC(C)C(=O)NC2CN(CC3CCN3S(C)(=O)=O)C2)ccc(F)cc1 c1(C(=O)NC2(CC=C)CN(C(C3CCCC(C(=O)OC)C3)=O)C2)cncc(Cl)c1C C1(NC(C2(CC(C)C)CC2)=O)(CNC(=O)COCc2cnsc2)CCC1 c1(OC)cn2c(cc1=O)CN(C(c1ncnc3c1c(Br)cn3C)=O)CC2 CCC(CC(F)F)C(=O)N1CC=C(CNC(c2cc(C(F)(F)F)ccn2)=O)CC1 CCC(CCC(=O)N(CCC(C)NC(c1ccc(CO)cn1)=O)C)OC C1(C)(NC(CCSC)=O)CCCCC1C(=O)NCCC1CCN(C)CC1 c1(C(N2CCC(N(C(=O)Cc3cccs3)CC)C2)=O)cccc2nc(O)ccc12 CC12CN(C(C3CCO3)=O)CC1(C)CN(C(c1cccn3ccnc13)=O)C2 O=C(NNc1ccccn1)C(F)n1cc(-c2ccccn2)nn1 C(=O)(C1=CC(C)(CC)C1)NC(CC)(C)CCNC(c1nocc1C)=O C1(CC(=O)NCC(=C)CCNC(c2ccc(Br)s2)=O)CCC(C)(C)C1 c1(COC)cc[nH]c1C(=O)NCc1ccc(C(=O)NC(C2CCOC2)CO)s1 c1(NC(C(=O)NCC(C)(CO)NC(C(F)=CC)=O)=O)ccc(OC)cc1 CC(CC(=O)NC1CCC(NC(=O)Cc2ccc(O)cc2)C1)CC(F)(F)F C1(C(=O)NC2(CC3CC3)CC2)CCN(CC(F)F)CC1.CC1CNC(=O)CNC1 C1(NC(CP(C)(C)=O)=O)COCCN(C(=O)COC2CCOC2)C1 c1(OCC)c(CC(=O)NC2CN(C(=O)C(C)CC(C)C)CC2C)cccc1Cl c1(CNC2(C(=O)NC3C(NC(=O)OC(C)(C)C)C3)CC2)cnc(N2CCOCC2)s1 c1(CC)cccc(C(=O)NC(CNC(C2(C)CC3CC3C2)=O)C2CC2)c1O C1(C(N(C)CC2(NC(c3cccnc3S)=O)CC2)=O)CC2CCC(C1)O2 N1(C(CCC=CC)=O)C2CCC1(CNC(c1cc(CC)on1)=O)CC2 Cc1cc(C(=O)NC2CC(NC(=O)OC(C)(C)C)C2(C)C)sc1Br.C(CO)N c1(C(=O)NCCC(C)NC(c2nnn(C)n2)=O)cnc(-c2ccccc2)[nH]1 N1(C(CSCC(C)C)=O)CCC2(CNC(c3cc(Br)c[nH]3)=O)CCCCC12 CC(C)C(C(=O)NCC(C)NC(=O)C(c1cccc(F)c1)O)C(C)C C1(NC(c2csc(Cl)c2)=O)CC2(CCCN(C(=O)C3=CSCCO3)C2)C1 N1(C(CCCCN(C)C)=O)Cc2nccn2CC(NC(C23CCN(CC2)C3)=O)C1 N1(C(C(C2CC2)NC(C=CC(=O)N(C)C)=O)=O)CC2(C=CCO2)C1 N1(C(C(C=C=C)C)=O)CCN(C(c2cc(C3(C)CC3)n[nH]2)=O)C(COC)C1 C(CNC(C1C=CCC1)=O)(CC(=O)NCC(O)C1(Cl)CC1)OC Cc1cccc2c1OCC2C(=O)NC1CCN(C(=O)CC(F)(F)C(C)C)C1 N1(C(c2csc(-c3cccnc3)n2)C(=O)NCC(F)F)CCc2ccc(Cl)cc2C1 C(c1cccc(OC(c2cncn2C(C)C)=O)c1)=CC.c12ccc(s1)CNC2 N1(C(C(C)CC(N)=O)=O)CC2CCCC2(NC(c2cn(C(F)(F)CO)nn2)=O)C1 CCCC(C(=O)N1CC(C(=O)NCC2CCOC2C)(CC)C1)OC c1(-c2cc(C)nn2C)cccc2[nH]cc(CC(=O)Nc3cc(C)c(F)c(C)c3)c12 C1(NCc2ccc(SC)cc2)CCCN(CC2CCNC2=O)CC1 N1(C(c2n(CC)ccn2)=O)CCC2(CC2)CC1C(=O)NCC1CC2CCC2C1 c1(NC(c2cccc(Cl)c2)c2n(CC)nnn2)ccc(OCC(C)C)nc1 C(C(C)(C)CC(=O)NOCC1CCOC1)NC(c1c(C)nc(C)n1C1CC1)=O N1(C(c2cc(C)sc2)=O)CCC12CN(C(=O)CN1C(C)CCC1C)C2 C1(C)(COC)CN(S(=O)(=O)NC2CCN(C(C)C(=O)N(C)C)CC2)O1 N1(C(c2c(C)nc(Br)o2)=O)CCC(NC(C2(n3cnnn3)CC2)=O)C(O)C1 C1(N(C(C2C(C(=O)NC(c3cn[nH]c3)C)C2)=O)C)CCC2(CC1)CC2 Cn1cc(OCC(=O)NCC2COC(CNC(=O)C(c3ccccc3)=O)C2)cn1 C#Cc1c[nH]nc1C(=O)NCC(C1CC1)NC(=O)CCNC(=O)CC1CCCC1 c1(CC(=O)N(C(CNC(C(Cc2ccc(C)cc2)C)=O)C)C)cn2ccsc2n1 c1(C(=O)NCCN(C(C)C)C(C2CCN2S(C)(=O)=O)=O)cc2cc(Cl)cnc2[nH]1 Cc1cc(C)n(-c2ccc(C(=O)NCC(O)CNC(C3C=CCC3)=O)cn2)n1 C1(NC(Cc2cnc(C)s2)=O)CCCC2CN(C(c3nccs3)=O)CC12 C1(O)(C(=O)NC(CC(C)NC(=O)C(C)(C)C2CC2)C)CCCCCC1 C1(C(N(CCN=[N+]=[N-])CC)=O)(CC)CCCN(C(c2csnc2Cl)=O)C1 CCC(C)C(=O)C(=O)NCC(C)C(N1CCNC(=O)C1CCO)=O N1(C(CC(C)(C)OC)=O)CC(NC(=O)CSc2ccc(C)cc2C)CC2(CC2)C1 c1(OCC)cccc(C(N2CC(NC(C3CCC(F)(F)C3)=O)C(C)C2)=O)c1 C#CCC(C)(C(=O)NCC1CCOCC1)NC(=O)CC(CN(C)C)CC c1(CC(N2CCC(CN(C)C(c3scnc3C(F)F)=O)CC2)=O)cc(F)cc(F)c1 c1(CC)cc(C(=O)NC2CC(OCC(=O)NCC(C)(O)C3(C)CC3)C2)n(C)n1 N1(C(c2cccc(CC#N)c2)=O)CCCC2(C1)CN(C(c1cccnn1)=O)C2 n1(CC(CNC(=O)CC2(CO)CCC2)OC)cc(-c2csnn2)nn1 C1(NC(C(CCC)N(C)C)=O)CC2CC1CC2C(=O)N(C)CC1CCN(C)CC1 C(=O)(C1CCc2ccc(Br)cc21)OCCCC(CC)C N1(C(c2c(C)scc2)=O)CCC2(CCOC2)C(CNC(C23CC(C)(CO2)C3)=O)C1 N1(C(c2ccc(=N)[nH]c2)=O)CCN(C(c2cocc2Br)=O)CC(O)C1 Cc1ccc(C)c(OCCC(N2CC=CC2CNC(C2CC(C)(F)C2)=O)=O)c1 N1(C(CCCCC=C)=O)CCC2(NC(c3ccccc3OC)=O)CCCCCC12 Cc1cn(-c2ccccc2)[nH]c1=NC(=O)N1CCOC(c2cn(CCO)nn2)C1 c1(OC(C)(C)C(=O)NCC2CC2NC(=O)CCn2cnnn2)ccc(Cl)cc1 c1(NC)ccc(C(N)=O)cc1C(=O)NC(c1nnnn1C(C)C)C1(CC#N)CC1 c1(CNC(CC(CC)C)C(=O)O)noc2c1CC(C)(C)CC2 Cc1ccc(CNC(N2CC(c3cccnc3)C2)=O)cc1Br N1(c2nc(-c3c(SC)ncc(C)c3)on2)CCc2c(ccc(Br)c2F)C1 N1(Cc2cccc(C)c2)CC2CN(C(c3ccc(I)cc3F)=O)CC12 C1(OC)CCC12CC(C(=O)NCCC1(NC(C3C(C)(C)C3(C)C)=O)CCCC1)C2 c1(C(C)OC(C2CC2(F)Cl)=O)cccc(Cl)c1F Cc1cc(Cl)ccc1C(=O)NC1CCCC(CNC(c2cn3c(n2)CCC3)=O)C1 Cc1c(C(N2CCC(CF)C2)=O)cccc1C1CC1.c12coc(c1)CNC2=O C1(NC(C2(C)CC(F)C2)=O)CC2(CCN(C(=O)CC3CC4CC4C3)CC2)C1 CCC(C)(C#N)C(=O)NC1CC(F)(CNC(=O)C(C(C)C)NS(C)(=O)=O)C1 Cc1cc([N+](=O)[O-])cnc1C(=O)NC1CCCC1CNC(=O)C(C)(C)C1CCC1 C(=O)(C(C(C)C)NC(C1CC(CC)C1)=O)N(CCC)CCNC(C1CCC1)=O c1(OC)cc(O)ncc1C(=O)NC(C)CCNC(c1ccc(SC(C)C)cc1)=O C1(NC(C2C(C)OCCC2)=O)CN(C(c2ccc(F)c(F)c2)=O)C(C)(C)C1 C1(NC(Cc2c(C)nsc2)=O)CN(C(=O)CCc2ccc(=N)[nH]c2)CCC1C c1(C(N(CC(C)(C)C)CC)=O)oc2c(OC)cc(C)cc2c1C N1(C(C(C(C)C)C#N)=O)CC2OCCN(C(c3csc(S(C)(=O)=O)c3)=O)C2C1 C(=O)(C(CC)C(C)C)N1C(C)(CCC(N2CCC(CC#C)CC2)=O)CCC1 NS(=O)(=O)CCCC(=O)NC1CC(NC(c2ccn3c2CCCC3)=O)C1 Cc1cc(CNC(C2(N(C)C(c3cccc(Cl)c3)=O)CC2)=O)oc1C c1(C(N2CCC(CNC(C3(CC#C)CCC3)=O)C2(C)C)=O)ccn2ncnc2c1 c1(C(C(=O)NC(C2CCOCC2)C2CC2)N(CC#CC)C)cc(C)ccn1 C1(C(=O)NCC2N(C(CCCC=C)=O)CC=C2)CC2(C1)CC(CO)C2 C1(C(CNC(C=CCCC)=O)(C)C)CCCCN1C(C1CC2(CSC2)C1)=O CC1CCN(C(c2csnn2)=O)CC1NC(=O)CC12CCC(C)(C1)OC2 C1(C(C)C)CN(C(=O)C(F)=CCCF)CCN1C(=O)C(C1CCOCC1)F Cc1nc(C(F)(F)F)ccc1C(=O)NC(C)CCCNC(=O)CC(O)C(C)C C1(NC(N(C)Cc2sccc2Br)=O)C(=O)NCC1(C)C CC1(C)CN(C(C2C=CCN(C(C3(F)CC=CCC3)=O)C2)=O)CCC1O C1(C(C)NC(CCSCC)=O)CCCN1C(c1cc(C(C)(C)C)c[nH]1)=O C1(C(F)(F)F)(NC(C2CCN(C(C(CN(C)C)(F)F)=O)C2)=O)CC2CCC1CC2 N1(C(c2n(C)c(O)nc2)=O)CCC12CN(C(=O)CCNS(=O)(=O)c1cccs1)C2 C1(C(=O)NCCn2c(C)nnc2)CC(F)CN(C(c2c(Cl)cccc2Cl)=O)C1 C(CNC(C1C2CCCOC12)=O)(CC(=O)NC1COC(C(F)F)C1)OC C(=O)(CC1OCC(C)(C)c2ccccc21)OCCOP(OCC)(=O)C(=O)OC c1(CC)ccnc(C(N2CC(O)(C(C)NC(=O)CCCN(C)C)C2)=O)c1 N#Cc1sccc1C(=O)NC1(CO)CCN(C(=O)CSc2ccc(F)cc2)C1 N1(C(CC2(CSC)CC2)=O)CC(C)CN(C(c2c[nH]ccc2=N)=O)CC1C N1(C(c2c(C(C)=O)nccc2)=O)CC2CCC1CN2C(c1ccccc1F)=O Cn1cnn(CC(N2CCC2C(=O)NC2(C)CC3(CC3)C2)=O)c1=O C1(CNC(=O)CC(F)F)C2CN(C(c3cccc(-n4nccn4)c3)=O)CC12 c1(-c2cnc(N(CCC)Cc3ccccc3)c(C)c2)ccc2c(c1)C(N)C(=O)N2 C(=O)(C1CCc2scnc21)NC1CCC(NC(C(C)Cn2ccnc2)=O)C1 C(=O)(C#CC1CCOC1)N(C)CC1OCCN(C(C2(SCC)CC2)=O)C1 C=CCCCCCC(=O)NC(Cc1cnn(C)c1O)C(=O)NCC(O)C(CC)CC N1(C(CCCc2onc(C)n2)=O)CC2CCN(C(=O)CCC(N)=O)C(C2)C1 Cc1cn2c(n1)CN(N1CCOC(CN(C)Cc3ccc(Cl)cc3)C1)CC2 C(C(CO)CC(C)C)NC(C1(CCNC(C(C=C)O)=O)CCCC1)=O N1(C(C(CC=C)CNC(=O)Cc2cccc(F)c2)=O)CCC2(CNC(=O)N2)C1 c1(OC)ccc2[nH]cc(C(C)CNC(=O)CC3CC(C)CC(C)(C)C3)c2c1 N=c1[nH]c(=NCC2CCC3(CC3)C2)[nH]c(=NC2CC(N3CCCCC3)C2)[nH]1 N1(C(CCCC#CC)=O)CC2=C(C1)CN(C(c1c(Br)ccc(C)c1F)=O)C2 C(=O)(C1(C)CCc2ccccc21)N1C(CN(C(CCN(CC)CC)=O)C)CCC1 C1(CNC(C(CC)C)=O)CCC2CN(C(=O)CSCC(=O)OC(C)(C)C)CC12 N1(C(C(C(C)C)C)=O)CC(C(=O)N=c2ccn(CC(N)=O)[nH]2)C(C2CC2)C1 Cc1c(C(N2CCC(C)(CCNC(C3C4COCC34)=O)C2)=O)cccc1N c1(C(=O)NCC2N(C(CCN(C3CC3(F)F)C(C)=O)=O)CC2)cccc(C#N)c1 CCC(CCC(=O)NCc1ocnc1C)NC(C1(C)CCN(C)CC1)=O CCC(c1ccc(C)cc1)=CC(=O)NCC1CC1CNC(=O)C(C)(C)CC(C)C C1(CNC(C=NOC)=O)N(C(=O)Cc2ccc(C3CCC3)cc2)CCCC1(C)C c1(C(N2C(CNC(c3cnco3)=O)CCC2)=O)ccc(C2CCCOC2)cc1 c1(CNC2C(COC)CCCC2)cccc(OC)c1F c1(OC)ccc(O)cc1C(=O)NCCCOCCNC(c1ccc(C#N)cn1)=O C(=O)(CC(C)CC(C)C)NCC(CC)(C)NC(=O)CNC(C1CCCCC1)=O Cc1cc(C(=O)NC2COCCC2NC(C2(C)CNC(=O)C2)=O)nc(N(C)C)n1 N#Cc1ccsc1C(=O)NCCCN(CCO)C(c1ccc(C2CC2)nc1)=O N#Cc1ccc(F)c(C(N2CCCCC2c2ccon2)=O)c1Cl c1(C(=O)NC(CCOC)CNC(=O)C(N2CCC(C)C2)=O)n[nH]c(C)c1O N1(C(c2nc(C)n(C)c2)=O)CCN(C(c2ccn(C3CC3)n2)=O)C(CF)C1 C1(C(=O)NCCCCCCC)CN(C(c2cnc(C)s2)=O)CCC1(C)C c1(C(N2CCC(C(C)C(=O)NC(C3(O)CC3)C)CC2)=O)cc(O)cc(F)c1 CP1(=O)CCN(CCCNC(C2CC2c2ccc(-n3ccnc3)cc2)=O)CC1 c1(SC)nc(N2CC3CCN(C(=O)C(C)(CO)CO)C3C2)c(Br)c(C)n1 Cc1ccc(C=CC(=O)NCC23CC2CN(C(=O)C(C(C)C)n2cnnn2)C3)o1 c1(N(CC(C)C)C)cc(C(=O)NCCCCNC(=O)CC2(C)CCCO2)ccn1 C1(C(=O)NC2(CC(=O)NCC3(C)CCCCO3)CCC2)CC2(CCC2O)C1 N1(C(c2ccc(C)nc2)=O)CCC2CN(C(=O)C=CC3CCCCCC3)C2C1 CCCC(C(=O)N(C1CCN(C(C2CC(=O)C2C(C)(C)C)=O)C1)CC)NC(N)=O CCC1=C(C(=O)N(C2CCN(C(C3(C(F)(F)F)CCC3)=O)CC2C)C)CCCO1 Cc1nn(C)c(C(N2CCC(CO)(CNC(=O)C3=CCCCC3)CC2)=O)c1Cl c1(NCC2CC(CNC(C3(n4cccc4)CCCC3)=O)C2)ncc(O)cn1 N1(C(c2ccn(CNC(COC)=O)c2)=O)CC2CCN(C)C2C1 C1(C)(C(=O)NC2CC(C)N(C(c3n[nH]cc3F)=O)CC2)CCC2(CC1)OCCO2 CC#CCCC(=O)N1CC2C(CNC(c3sc(Br)nc3C)=O)C2C1 C1(C2(O)CCN(C)CC2)(C(=O)NC(COc2ccc(C)c(C)c2)C)CC1 N1(C(CCc2cc(C)[nH]n2)=O)CC2CCC1CC2NC(=O)Cc1cc(C)oc1C C(=O)(CC(F)(F)C(F)F)NC1CC(NC(=O)Cc2cc(Br)ccc2O)C1 c1(NC(c2nnnn2CCC2CC2)CCSC)ccc2c(c1)C1CCC2N1 C(=O)(CC(F)(F)C(F)(F)F)N1CCN(C(C(C(C)(C)C)=O)=O)C2C1C2 CCCC(C)(O)C(=O)N1CCCC(C)(NC(C2(c3cc(C)cc(C)c3)CC2)=O)C1 C(=O)(CCC(=O)NC(C(=O)NC(C)CF)C1(C)CC1)NC n1(-c2ccc(C)cc2)cnc2c1CCN(N1CCCN(C3CCC3)CC1)C2 c1(OCC)cc(C(N2CC(C(C)NC(=O)C(CC(C)C)OC)C2)=O)ccc1OC n1(CC)nnc2cc(C(N3CCC(NC(=O)CC(C)F)C34CCC4)=O)ccc12 C(=O)(C(CC)(CC)CC)N(C)CC1CCN(C(c2cccc(CC)c2F)=O)C1 C1(C(N(C)CC2CN(C(c3ccn(C(F)F)n3)=O)CCO2)=O)CCCCCN1C CC(C)C(O)C(=O)NC(C)CCCNC(C1(OCc2ccccc2)CC1)=O C1(CN(C)C(c2ccco2)=O)CN(C(c2cc(Br)n(C)c2)=O)CC12CC2 Cc1cc(C(=O)NC(c2c(C)cccc2Br)C)cc(Br)c1 C#CCCCCCCCC(=O)NCC(CO)NC(=O)C#CC1(C)CCCO1 Nc1ncc(Br)cc1C(N1CC(NC(=O)CCc2cnn[nH]2)C(O)C1)=O N1(C(COCCC(C)C)=O)CSCC1C(=O)NCC1CCN1C1CC1 N1(C(C=CCOC)=O)CSCC1C(=O)OC(C)(C)C.C1(C=O)CC(CF)C1 N1(C(CCC(=O)OCC)=O)CC2CC1CN(C(c1ccc3c(n1)CCC3)=O)C2 N1(C(C2N(C(Cn3c(C)nc(C)n3)=O)CCC2O)=O)CCCC(C)C1CO c1(CNC(C(=O)NCC)=O)cccc(C(N2CCC(CF)C2)=O)c1 CCCCCCC(C)C(=O)N(CC(C)N(C(=O)C(COC)N(C)C)C)C c1(N2C(C)(CNC(COc3cccc(C)c3)=O)CCC2)ncc([N+](=O)[O-])cc1Cl N#CC1(C(=O)NC2CC(OCC(=O)Nc3cccc(CO)c3)C2)CC2CCC1C2 N1(C(Cc2ccn(C)n2)=O)CCC=C(C(=O)N(c2cnc(O)nc2O)CC#N)C1 c1(N2CCC(C(=O)NCC(C)N(C)C(C3C=CC=CC=C3)=O)C2)ccccc1F C(=O)(CS(=O)(=O)c1ccccc1F)NC(CNC(C1(C#N)C(C)C1)=O)(C)C N1(C(c2ccc(CCC)cc2)=O)CCC(C(=O)OC)CC1C(F)(F)F Cc1ccc(C(=O)NCC(CNC(C2CCS2(=O)=O)=O)CO)nn1 c1(OCC2CC(OC)CN2C(=O)OC(C)(C)C)ccc(Br)c(C(=O)CN(C)C)c1 C12(NC(CS(CCC)(=O)=O)=O)CC(C)(C1)OC21CN(C(=O)COC(C)CC)C1 C1(C(=O)NCCC2CCCN(C(C(CO)OC)=O)C2)CCCCCN1C N1(C(C(C)SC(F)(F)F)=O)CCC(C)C(NC(=O)CCCN2C(=O)CCC2=O)C1 C(=O)(CCCCCNC(=O)C(C1CCCCC1)=O)NCCCc1n(C)cnn1 CC1(NC(C23CCC2C3)=O)CN(C(=O)COCCN(C)C)C1 CC1C(NC(=O)CC23CCC(CC2)C3)CCN1C(c1cccc(C(C)(F)F)n1)=O c1(C(=O)NCC(CNC(CCC(=O)NCCCOC)=O)O)ccc(Cl)c(O)c1 O(NC(=O)CC(C)NC(c1c(C)cnnc1O)=O)C(C=C)C N1(C(Cn2c(CCC)nnc2S)=O)CCN(C(c2ccc(O)nc2)=O)CC(O)C1 c1ccc2c(=NCCCC3CCOC3)[nH]c(=NCC3CCCCO3)[nH]c2c1 N1(C(C(F)OC)=O)CCCC1C(C)NC(=O)C(O)c1ccsc1 N1(C(C2CCCN(CCC)C2)=O)CCOC2CN(C(=O)CC(=O)NCC)CC12 C12(C(=O)OCC)CCCC1CN(C(c1ccc(C)c(I)c1)C(=O)NCCC#N)C2 C(=O)(C1(C)CCn2c(C)nnc21)N1CCC2(CCN(C(c3c(C)snc3)=O)C2)C1 CC(C)C(C)C(=O)N1CC(C(O)C(=O)NC2CC(N3CCCC3)C2)C1 c1(C(=O)NCC(C)(C)NC(CCc2c(C)ncnc2O)=O)cc2n(n1)CCOC2 C1(CNC(c2ccc(CO)c(F)c2)=O)CC2CCC1N2C(C1CCCCO1)=O C1(CNC(c2c(CC)cco2)=O)CN(C(=O)C(C)(C)O)CC1O N1(C(c2c(C)nc(C(C)(C)OC)s2)=O)CCN(C(=O)CS(C)(=O)=O)C2CC12 C1(CC(C)NC(=O)CC2(O)CCCC2)CCN(C(C2CCCCCC2)=O)CC1 C1(OCCC)CCCN(C(C2CCC(NC(c3cnn(C(F)F)c3)=O)CC2)=O)C1 C1(NC(C(C)NC(=O)C(C)(C)C)=O)CN(C(C2CCC2)=O)CC1O C(=O)(C(C)CCNC(=O)C(CC1CC1)NC(C12CCC(C1)C2)=O)OC n1(CCC)ncnc1CNC(C1CC(N(C)C(c2cc(CC)on2)=O)C1)=O c1(OC)cc(F)c(S(=O)(=O)NC(c2cc(C)c(=O)n(C)c2)=O)cc1OC CC1(C)CC(S(N)(=O)=O)CN1C(c1cc(C(F)(F)F)cc(Br)c1)(C)C N1(c2snc(COC)n2)CCC2(CC1)CC(NC(c1cnnc(Cl)c1)=O)C2 CC1OC2(CO)CC1(C(=O)NC1CCCCN(C(C3(CO)COC3)=O)C1)C2 C1(NC(C2COCCO2)=O)CCN(C(c2ccc(-c3ccccn3)o2)=O)C12CC2 C1(C(=O)NCC2C(CC(=O)NC(c3nc[nH]n3)CC)C2)CCCN1C(=O)C1CC1 Cn1cnnc1CCCC(=O)NCC1CCC(NC(=O)CC2(C)CC2(Cl)Cl)C1 c1(CC)ccc(C(=O)NC(C(N2CCC(OCC(C)C)C2)=O)c2ccco2)cc1 N1(C(CN(C(COC)=O)C)=O)CC(C)(C)CC1CNC(c1cn(C)nc1SC)=O N1(C(Cc2c(C)cnn2C)=O)CCCC(F)(C(=O)NCCc2nnc(C)n2C)C1 N1(C(CC=CC=C)=O)CC2CC2(CNC(C2CSCN2C(C2CCC2)=O)=O)C1 c1(CC(=O)NCC(C)NC(CCCNC(=O)NCC#C)=O)cccc(Cl)c1 n1(CC)ncc(Cl)c1C(=O)N(C)CC1CN(C(C2COC2)=O)CCO1 C1(NC(C(CC)n2ccc(C3CC3)n2)=O)CCCC(CNC(c2cnns2)=O)C1 Cc1cc(NC2CC(C)N(C(c3ccn(CC4CC4)c3C)=O)C2)n2ncnc2n1 c1(C(=O)NCC(=O)NCC2N(C(C(CC)C)=O)CCCC2)cccc2[nH]ccc12 CC1C(C(=O)NC2(C(=O)N(C3CN(C(C)C)C3)C)CC2(C)C)=NOC1C N1(C(CCC#C)=O)CC2(COC(CNC(=O)C(C)CN3CCOCC3)C2)C1 CCC(C)(COCC(=O)NC1CCC(C(F)(F)F)CC1)CNC(=O)OC(C)(C)C N1(C(C(C2CCCC2)OC)=O)CC2CCC(CNC(C3CCOC3)=O)(C2)C1 N1(C(C2(OC)CCOC2)=O)CC(C(=O)NC2CCC(C)(C)C2)CCC1(C)C c1(C(=O)OCC)ccc(C(=O)NC2CCC(N(C)C(c3ccc(C)o3)=O)C2)cc1 CC1(C)CN(C(c2cc(N)cc(O)c2)=O)CCC1NC(C1CCCC2(CC2)C1)=O c1(C(N(C(CCNC(Cc2ccn(CC)n2)=O)C)C)=O)nccc(C)n1 N1(C(CN(C2CCS(=O)(=O)C2)C)=O)CCC(F)(CNC(=O)C2=C(Cl)CC2)C1 C#CCCC(O)C(=O)N1CCN(C(=O)CCc2cnc(O)[nH]2)CC1CO CC(CCC(C)(C)C)C(=O)N1CC2(C(=O)NC(C(O)CO)C3CC3)CCC1CC2 c1(C(=O)NCC(COC)NC(=O)CCc2cnn[nH]2)ccnc2ncccc12 C1(CN(C(c2nccs2)=O)CC)CCN(C(=O)C(C2CCC(=O)N2)C)CC1 C1(C(N(CC(C)NC(=O)CC2(C)CCCCC2)C)=O)COCC(C)(C)O1 c1(C(=O)NCC2N(C(CCCN(C(C)C)C)=O)CCC2C)cn2c(n1)COCC2 C1(F)(CNC(c2cn(CC(N)=O)nn2)=O)CCC(CNC(=O)C=CC2CC2)C1 N1(C(C(CSC)C)=O)CCN(C(=O)CSS(C)(=O)=O)CCC1C N1(C(CCOCCCNC(c2ccn(CCC)n2)=O)=O)CC2OC(=O)N(C)C2C1 C=CCC(C(=O)NC1CC1c1ccnn1C)NC(=O)COC1CC=CC1 C(CNC(C12CSCC1C2)=O)(CC(F)(F)F)NC(C1C2COCC12)=O n1(C(CC)C)ccc(=NC(=O)C(C2CCCO2)N(C)C(=O)OC(C)(C)C)[nH]1 c1(CNC(c2cnc(CC)[nH]2)=O)ccc(CNC(=O)Cc2cnoc2)cc1F O=C1CC(NC(=O)CCC2CCCN2C(c2ccc(Cl)cc2)=O)CN1O N(C(=NCCC1CC1)NC(C)(C)CF)CC(C)OC c1(C(=O)N(C2(C(=O)NCCC3(CO)CCC3)CCC2)C2CC2)occ2c1CCC2 c1(C(N2C(CC(=O)NCCC(=O)OC)CCC2)=O)c[nH]nc1[N+](=O)[O-] N1(C(c2ccccc2-c2ncc[nH]2)=O)CC2CC(NC(C3CC(O)C3)=O)CC1C2 N1(C(C2(C)CCNC2=O)=O)CC23CCCC2(C1)CN(C(=O)Cc1ccno1)C3 Cc1ccc(C(N2CCC(C)(NC(c3cccc(-n4ccnn4)c3)=O)C2)=O)n1C C1(CCCNC(C(C)OC)=O)CN(C(=O)C(C)C2CC2(Cl)Cl)CC1n1ccnn1 C1(NC(c2cc(C)sc2C)=O)C(C)CN(C(c2ccnc(C3CC3)c2)=O)CC1C N1(C(C2(C)CCN(C(C)=O)C2)=O)CC(NC(C2CCCO2)=O)C2CC2C1 C1(C(=O)OC)(CO)CCCN1C(=O)NCc1cc(C)cs1 c1(NCC(CO)Cc2ccc(Cl)cc2Cl)cc(=NCC2CSC2)[nH]cn1 c1(C(=O)NCCC2CN(C(C=C(CC)C)=O)C2)sc(S(N)(=O)=O)c(C)c1Cl O(S(=O)(=O)C1CC12CCC(=O)CC2)c1cc(Br)cc(C)c1O N1(C(CC=C)=O)CCCCC(N(C(=O)CCCCN2C(=O)CCC2=O)C)C1 N1(C(c2c(OC)nccn2)=O)CCC(O)C2(CCN(C(=O)CC3CCC3)CC2)C1 C1(OC)(CNC(C2(C)C=CCCC2)=O)CCN(C(c2cccc(N)c2F)=O)CC1 C1(NC(=O)NC(C)C(C)n2ccnc2)CCN(c2ccnc(Cl)n2)CC1 N1(C(C(CC(C)C)ONC(c2cc(C#N)c[nH]2)=O)=O)CCC12CCCSC2 c1(C(=O)NCCNC(C2CC(Cl)(Cl)C2)=O)cc2ccncc2s1 NS(=O)(=O)CC(=O)NC1CC(NC(C2CCCN(C(c3ccccn3)=O)C2)=O)C1 C#CC1CC2(CC2)CN1C(C1(CNC(C2CCN(C)CC2)=O)CCCCC1)=O C(=O)(C(O)C(CCC)NC(c1c(C)nn(CC)c1C)=O)NCCCCC#C N1(C(c2c(C)ocn2)=O)CC(C)CCC1CNC(c1csc(C(C)(F)F)n1)=O C1(NC(c2cnc3n2CCC3)=O)CC2CN(C(=O)CN3CCCNC3=O)CC12 N1(C(COCCN(C)C)=O)CCCC(C(=O)N(C2CC(C)(C)C2)C)CC1 CCC(C(=O)N1CCSCC1CCNC(c1n[nH]c(C)n1)=O)C(C)O C1(C(N(C(C=C)C2CC2)C)=O)CCN(C(=O)CC2CC(=O)C2)CCO1 CCCCC#CC(C)(C)NC(=O)CCN(C(=O)CCOC(C)C)CCO C1(NC(CC2(CNC(C(C)c3ccsc3)=O)CC2)=O)CC(O)C(O)C1 c1(C(N(CCNC(COCCC=C)=O)CCOC)=O)sc(Br)nc1C CCCC(C(=O)N1CCC(C(=O)NCC(F)(F)CO)C(C)(C)C1)C(C)C c1(CCNC(=O)NC(C)C(N2CCCCCC2)=O)cccc([N+](=O)[O-])c1 CON1CC(C(=O)NC2CC23CC(NC(c2ncnc(C)c2C)=O)C3)CC1=O c1(C(N(C)CCOCC2CC2)=O)cc(Cl)ccc1N1CCCC1 C1(C(N2CCN(CCC)CC2)=O)CN(C(c2ccncc2F)=O)CC1(F)F c1(-n2c(C)nnc2)ccc(C(=O)NC(C)(CNC(c2cscn2)=O)CO)cc1 c1(CC)nc(CC(=O)OC(=O)CCc2nc(C3(OC(C)(C)C)CC3)no2)cs1 C1(CNC(CC2(C(=C)F)CCC2)=O)CC2(CCC2)CN1C(c1cscc1C)=O CC(C)C(C)CN=c1[nH]c2c(c(=NCc3ccc(C(N)=O)cc3F)[nH]1)COC2 CCC(CCCC(=O)NC(C1CCOC1=O)C)NC(c1c[nH]c2cccnc12)=O Cc1cc(C#N)ccc1C(=O)NCCC1CCN(C(=O)CSS(C)(=O)=O)C(C)C1 c1(C(=O)NCC(c2ccncc2)C)ccc(N)c(F)n1 N1(C(c2c(C)noc2C)=O)C2CCC1C(CNC(c1nsnc1O)=O)C2 CC(CN(C(c1ncccc1Cl)C(=O)N(C)C)C)C(F)(F)F.C12CC(C1)C(=O)N2 N1(C(C(CC)C)=O)CC2(CC2)CC1C(=O)N(C)Cc1cnc(C)cn1 C1(C(=O)OC)CN(CC(=O)NC(=O)Nc2c(C)cc(Cl)cc2Cl)CC2(CC2)C1 c1(-c2n(C)ncc2NC(=O)CC2COC3CC2C3)ccc(F)cc1F c1(C(CNC(c2cccc(OC)n2)=O)NC(C2CC(O)C2)=O)ccc(F)cc1F c1(C(=O)NC2CN(C(C(C)(F)F)=O)C2)cncc(COC(F)(F)F)c1 C1(C2CC2)(CNC(C2CCN(CCF)CC2)=O)CCN(C(=O)COCC2CC2)C1 C(=O)(CC(C)CF)NCC1CC(CNC(c2ccc(CN(CC)CC)o2)=O)C1 C(=O)(CCCCCN=[N+]=[N-])N1C(C)CC(NC(=O)CCOC2CCCCC2)CC1 C(=O)(CC(C)C(=O)N1CCCN(CCNC(=O)C(O)CC(N)=O)CC1)OCC CC1CN(C(=O)C=CS(C)=O)CCCN1C(c1cccc2nonc12)=O C1(C(=O)NCC(CNC(c2ccc(CN(CC)CC)o2)=O)O)COCCOC1 c1(OCC=C)ccccc1CN1CC2(CC2C(N2CCCCC2C(N)=O)=O)C1 C1(C(=O)NC2CC3(CN(C(C(CC)C(=O)OC)=O)C3)C2)Cc2cc(C)ccc2S1 c1(CC(N2C(C(=O)NCCCn3ncc(C)c3)CCC2)=O)cnn(C)c1C Cc1c(O)ccc(C(=O)NCC2CCN2C(=O)C(C2CCCCC2)C)c1C CCC(C)C(CNC(=O)C(COC)NC(=O)C(C1CCCCC1)O)CO N1CC=C(CC(=O)N(C)CCOC)CC1.C(CCCCC=O)OCCOCCOC C1(C(N2CC3CN(C(C(C(C)C)O)=O)C3C2)=O)CCCC2CCCCC12 c1(C(=O)NC2(CC=C)CN(C(c3csc(O)n3)=O)C2)ccc(C)c(Br)c1 CP(C)(=O)CC(=O)NCCC1(O)CCN(C(=O)Cc2ccc(O)cc2)C1 N1(C(COC)=O)CCCC1C(=O)NCC1(C(=O)OCC)CCC1 c1(SCC(=O)NCC(CNC(=O)C(C)Cc2ccncc2)OC)ccc(Cl)cc1 C(=O)(C(CCOCCO)NC(C1CC(C)(C)C1)=O)NCC#CC C=CCC(CC)C(=O)N1CCOC(CNC(=O)C(CC2CCCCC2)C(C)C)C1 c1(C(=O)NCCN(C(C(CC(C)C)O)=O)C2CC2)ccc2ccn(CC(F)F)c2c1 CN=c1ccc(C(N2CC(CC(C)(C)CNC(c3cc(C)nc(O)c3)=O)C2)=O)c[nH]1 Cc1ccc(S(C)(=O)=O)cc1C(=O)NCCC(C)N(C)C(c1[nH]c(O)nc1C)=O c1(CCC(=O)NCC2CCCN(C(c3n(C)c(O)nc3)=O)C2)ccc(Cl)c(Cl)c1 Cc1n[nH]c(C)c1CC(C)C(=O)NC(C1CCCC1)CNC(=O)C(F)F C=CCCC(C)(C)C(=O)N1CC2(CNC(C3CCCC3OC)=O)CC1CCO2 Cn1ccc(C(=O)NCCC2(O)CN(C(=O)C(C)(F)CC3CCCC3)C2)cc1=O Cc1ccc(C(=O)NC2CCCC2CN(C)C(C2CCCOC2C)=O)cc1C c1(C(C(=O)NCCC)N(C(C)CS(=O)(=O)CC)CCF)ccc(Cl)cc1F c1(CN2C(C(=O)NC(c3ccccc3)CC)CCCC2)ccc(OC)c(OC)c1 CCC(CCCC(=O)NCC(C)(C)C(C)C)NC(c1ccc([N+](=O)[O-])[nH]1)=O N1(C(Cc2cccc(C)c2)=O)Cc2occ(C(=O)NC3CCCCC3F)c2C1 CC(C)CCCC(=O)NC1C=CC(CC(=O)NCCC(C)CO)C1 C(=O)(CCCC1CCCC1)N(CC(C)NC(=O)CSC1CCOC1=O)C1CC1 c1(OC)ccc(C(C)(C)NC(C23CC(n4cc(CC5CC5)nn4)C2C3)=O)c(F)c1 C1(C(=O)NCC2CC(NC(c3c(C)ncn3C)=O)C2)CCC(=O)N2CCCC12 CC(C)(CC1CCC1)C(=O)N1CCC(NC(C2CCNC2=O)=O)C1 c1(C(=O)NCC(C)NC(=O)CC2CC3CCC2CC3)cc2c(nc1O)CCCC2 C(CN=c1nc(CC)cc(C)[nH]1)(C(C)(C)C)NC(c1cc(CCC)[nH]n1)=O C1(C(N2CCC(N(C(=O)CN3CCC(O)CC3)CC)C2)=O)CCCC2(CC2)C1 N1(C(C2(CC)CCC2)=O)CC2(CNC(=O)CCC3CC3(C)C)CCC1CC2 c1(CN(C)C)cccc(C(=O)NCCCN(C)C(c2c(Cl)csc2Cl)=O)c1 CC(CNC(c1ccc(O)c(F)c1)=O)C(F)C(=O)NOCC1CCCC1 CCCCCCC(=O)N(C1CN(C(c2cccc(OC)n2)=O)C1)C C1(NC(CN(C2CC2)CC)=O)CCN(C(=O)CCc2nncn2C)CC1C(N)=O C12(C(=O)NCC3CCC(F)(CNC(CNC(=O)NC)=O)C3)CC1COC2(C)C N1(C(c2cc(CC)sn2)=O)CCC2(CC1)CC2C(=O)N(C)CC1(N(C)C)CC1 c1(OC)ccc([N+](=O)[O-])c(C(N2CC3CC2CN3c2ncc(C)c(C)n2)=O)n1 C1(CCC)CN(C(C2(C#N)CCCC2)=O)CC1NC(=O)C(c1ccccc1)C c1(C(=O)NCC2C(NC(c3cc(CC)[nH]n3)=O)CCC2)ccc2c(c1)NCCC2 C(C(C)(C)CC(=O)NC(CO)C(C)O)NC(c1cc(C(C)C)no1)=O CCCCCCC(=O)N1CCC(NC(C2COCCN2C(C)=O)=O)C1 c1(OC)c(C)cc(C(=O)NCC2CN(C(=O)CC3CN(C)C3)CCO2)cc1Cl c1(N2CCC(C(=O)NCCC)CC2)nc2ccsc2c(=NCC2CC2(Cl)Cl)[nH]1 C(C(O)CC(=O)NCCCC1(Nc2cc(C(F)(F)F)ncn2)CC1)N(C)C O=S(=O)(CCN=c1[nH]c(=NCC2CC2Cl)[nH]c2c1COC2)N1CCCCCC1 c1(NC(=O)CC2CCN(Cc3csc(Br)c3)C2)ccc([N+](=O)[O-])nc1 C1(c2nnnn2C2CC2)(NC(c2cccc(F)c2)=O)CCC2CCC1O2 C1(C(=O)NC2C3CC2CN(C(=O)CCC2CCCOC2)C3)CCN2CCCC2C1 CC(C)CC(C(=O)NCCN(C(c1cc(Cl)cs1)=O)Cc1ccccc1)N(C)C n1(C(C(=O)OCC)C)ccc(=NC(=O)C2CCCCC2CC)[nH]1 c1(C(N2CCC(N(C(C(CCC)O)=O)C)C2)=O)cccc2c1OCC(=O)N2 c1(C(C(=O)NC2CCOCC2)N(CCCOC)C)ccc(Cl)c(SC)c1 c1(-c2cccc(NC(c3ccc([N+](=O)[O-])cc3)=O)n2)ccc2ccoc2c1 C(c1cnn(C)c1C)=CC(=O)NC1C(SC)CN(C(=O)CS(N)(=O)=O)C1 C=CCCCC(C(=O)N(CC(C)O)CCF)NC(=O)COCC(F)F C1(NC(C2(CC)CC2)=O)CCCC1CNC(C1CC12CCC2)=O n1(CC(=O)NC23CCN(C(c4c(CC)scc4)=O)CC2C3)cc2ncccc2n1 C(C(C(=O)N1CC(n2ccnn2)C1)n1cc(C2(C(=O)O)CC2)nn1)OCC Cc1cc(C(N2CCN(C(=O)C(O)C3CCC3)C(C3CC3)C2)=O)c(Br)c(C)c1 N1(C(CSCCCn2c(C)nnn2)=O)CCC(F)(c2ccc(F)cc2)C1 N1(c2ccnc(C(CC)C)n2)CCC2(NC(C3CCCC(F)C3)=O)CCCC12 C1(NC(=O)NCC2(C)CCCCC2CO)CC2(CNC(=O)O2)C1 N#Cc1cc(Cl)c(Cl)cc1NC(C1CCCN1C(=O)CCNCc1ccc[nH]1)=O c1(C(N2CCC(CC(C)NC(C3CC4CC4C3)=O)CC2)=O)ncnc2cc[nH]c12 N1(C(C2CCC(C(=O)OC)O2)=O)CC(NC(=O)CC2CC=CCC2)C(C)C1 C=CC1CC(NC(=O)C(CCOC)NC(=O)CCN(C)CCO)CCO1 C1(CNC(C(C)NC(=O)NC)=O)CCc2cnnn2C1 N1(Cc2cnc(C(C)C)s2)CC2CC1C2C(=O)Nc1cncc(Cl)n1 O=C1CSCC(C(=O)NCC2(F)CN(C(C3CC(N4CC(O)C4)C3)=O)C2)N1 C1(NC(c2cccc(CC)n2)=O)CC(C)CN(C(=O)Cn2nccc2C)C1 N1(C(C2C(C)(C(C)C)C2)=O)CC(NC(=O)CN2CCOCC2)C(F)C1 N1(C(CNC(CC)=O)=O)CCCCC1C(=O)NCC=CC(C)(C)C c1(CC(=O)NCC=CC(=O)NCC2(C)N=C(C)SC2)cccc(C#N)c1 c1(C2C(C(=O)NCC(CNC(c3ocnc3C)=O)OC)C2)ccn(C)c1 C1(NC(=O)CCc2cnccn2)CN(C(=O)CSc2nncs2)CCC12CCC2 CC#CCCCC(=O)N(C1CCCN(C(c2c[nH]c(=N)nc2C)=O)C1)C Cc1cc(C(=O)NCC2(C)CCN(C(=O)C(C)(C)C(C)O)CC2)c(Cl)cc1F C1(C(=O)NC23CC(CC)(C2)C3)CC2CC1CN(Cc1ccc(OC)c(OC)c1)C2 C1(SC)CCN(C(C2CCC23CCC3)=O)CC1 c1(OC)ccc2c(c1)CC(C(=O)NCCCCNC(c1csc(Cl)n1)=O)CC2 Cc1cnn(CCCNC(c2nnnn2Cc2cccs2)(C)C2CC2)c1 c1(C(=O)Nc2nnc(CS(C)(=O)=O)s2)cc(OCC(F)(F)F)ccc1O c1(OC)ccc(N)c(C(=O)NCC(C)CNC(=O)CCc2cnn[nH]2)c1 N(C1c2ccccc2CC1NC(=O)CCC1NC(=O)NC1=O)C(C(C=CC)O)=O c1(C(=O)NC2(CCCNC(C(C)=C3CC3)=O)CC2)cncc(N(C)C)c1 CC(O)(CNC(=O)CC1CCCCN1C(c1ccsn1)=O)C(F)F c1(CNC2C(C)(C)C2)nc(Cc2ccccc2)cs1 C(CCC(C)C(=O)NC1CCN(C(C2CCC(=O)NC2)=O)C1C)OC C(=O)(C1=CCC(F)(F)CC1)N1CCC(CN(C(c2cn(CC)nc2C)=O)C)C1 S(=O)(=O)(C1=C2CCN=C2N=NC1)Nc1ccc(C)c(OC2CCOC2)c1 N1(C(Cc2ccc(C)o2)=O)CCCC(C)(CNC(C2CC(C(C)(C)C)C2)=O)C1 C(C(C)(CC)NC(C=CC(C)(C)NC(=O)CCOC1COC1)=O)SC Cc1ncc(C(=O)NC(CNC(c2cnn(C)c2)=O)C2CC2)n1C c1(C(=O)OCC)ccc(S(=O)(=O)NCC2(Cc3ccccc3)CCOC2)c(Cl)c1 C1(NC(C(C)NC(C2CCC2)=O)=O)CCOCC1NC(=O)Cc1ccccc1F C(=O)(C(C)(C)CC(C)C)NCC(CC)(CC)NC(=O)CCc1ccc(O)cc1 C=CC1(C(=O)N(CCCCCC(=O)Nc2cccnc2)C)CCCCC1 C1(C(N2CCC(Cn3cc(-c4cccc(C)n4)nn3)C2)=O)CCCC(=O)CC1 Cc1ccc2nsnc2c1C(=O)NCC1(C)CCCN(C(=O)C=CC=C(Cl)Cl)C1 C(=O)(CCCCCN(C(=O)Cc1ncccc1F)C)N1CC(C)(CC)C1 c1(C(N(C2CCCN(C(C34C=CC(CC3)C4)=O)C2)C)=O)cc2nc(F)ccc2o1 C1(C(=O)NC2CC(NC(C3CCC(O)C3)=O)C2)CCN(c2cc(O)ncn2)CC1 c1(C(=O)NC(CNC(C(C)(C)CF)=O)C2CC2)snc2ccccc12 C1(NC(C(CCSC)OC)=O)CN(C(c2nc[nH]c2C(F)(F)F)=O)CCC1F C1(C(=O)Nc2cn(C)nc2)(CNC(c2cccc(CO)n2)=O)CC(C)(C)C1 N1(C(c2nc(C)c(Br)cc2)=O)CC2(CCC(NC(=O)C(=O)NC3CC3)C2)C1 c1(-n2c(C)ncc2)cccc(C(c2nnnn2C)(C)NCCN2CCOC(C)C2)c1 c1(CN=C(NC(C2CCCO2)C)NC2CC(C3(F)CCC3)C2)cccc2c1OCC2 N1(C(CCC2(C)CC2)=O)CCC2(NC(=O)OCc3ccccc3)CC2C1 CC1(C(=O)O)CC2CC2C1.c1(-n2cc(C34CN(C3)C4=O)nn2)c[nH]ccc1=N CON(C)CCCNC(C1CC(O)CN1C(c1c[nH]nc1C1CC1)=O)=O C1(C(N2C(CNC(Cc3c(C)non3)=O)CCCC2)=O)CC2(CCC2O)C1 N1(CC(=O)NC2(C(=O)Nc3ccnc(-n4cncn4)c3)CCC2)CCC(F)(F)C1 C(=O)(C(F)(F)C1(O)CCC1)NCCC1CC(NC(C(c2cscn2)N(C)C)=O)C1 C(=O)(N=S1(=O)CCCC2(C1)OCCO2)N1C2(CN)CC(C1)C2 Cc1cccc(C(N2CCC(NC(=O)CS(=O)(=O)N3CCOCC3)C2C)=O)c1C c1(C(N2CCNC(C(=O)Nc3ccc(O)c(CO)c3)C2)=O)cc(Br)cc(F)c1O C1(CNC(C(C)C2CCCO2)=O)CCN(C(=O)CC)CC1.C12(C)CC(C1)C(=O)N2 C1(NC(C2CCC(NC(=O)C=CC3CCCC3)C2)=O)CCc2nncn2C1 N1(C(C2(C#N)CCCC2)=O)CCC(C2CCN(C(=O)C(F)(F)c3nccs3)C2)C1 C#CC1CN(C(=O)CNC(=O)CNC=O)CCN1C(C1CSC1)=O C1(CNC(CN(C(C2C(CCOC)C2)=O)C2CC2)=O)CC2CCC1O2 c1(OCC)nc(C(N2CCCC2C(C)NC(=O)C(C)Cc2ccccn2)=O)co1 CN=c1ccc(C(=O)NCC(CO)NC(=O)COc2ccccc2C)c[nH]1 N1(C(CC(CC)C2CC2)=O)CC2CC1CN2C(C12CCC(C1)OC2C)=O C(=O)(C(F)(F)C(F)(F)F)NC(CCC)CC(=O)NC1CC(OC(C)C)C1.OCC C1(C(=O)Nc2c(C)onc2Br)C2CC(C(O)C2O)S1(=O)=O c1(C(=O)NCC(=O)NCC2(O)CN(C(C(CC=CC)C)=O)C2)cc(C)cc(C)c1 C1(CCC)CN(C(C2CC(O)CN2C)=O)CCN1C(c1nc(C(C)C)oc1C)=O c1(-c2nc(CC)nn2C)ccc(-c2nccs2)cc1F CCCC(CC)CCC(=O)N(C(C)C(=O)Nc1cc(C)cc(C)c1O)CC N1(C(C2N=C(C)SC2)=O)CCCC(NC(c2cc(C)c(O)nn2)=O)C1C c1(OCC)ncc(C(=O)NCC=CCNC(C2COC(=O)C2)=O)cc1Cl Cc1cc(C=CC(N2CC(CNC(c3cn(C)cn3)=O)C(C)C2)=O)on1 C1(NC(C(CC)(C)F)=O)COC2(C1)CN(C(c1cc(CC(C)C)nn1C)=O)C2 c1(C(N(C)CC2(NC(C3COCCC3(F)F)=O)CC2)=O)ccc2cccnn12 C1(NC(c2snc(Cl)c2Cl)=O)CC2CCC1N(C(=O)C1=CCCCC1)C2 N1(C(C2C(C)CC=CC2)=O)CC(C2CN(C(=O)Cn3cnnn3)C2)C1 N1(C(CCC(=O)NCC)=O)CC(NC(C2CC2c2cccs2)=O)CC2(CCC2)C1 N(C(=NCCc1sccc1C)NCC1CC(C)(F)C1)C(C=C)C c1(CC(=O)NCC(CNC(c2c(C)nco2)=O)C(F)(F)F)nc2c([nH]1)CCCC2 CC(C)C(C(=O)NCCNC(c1cn(C)nc1C1CCCCC1)=O)NC=O c1(C(=O)NCCOC2CN(C(C3(CC#C)CCCO3)=O)C2)ccc(Cl)cn1 CCCCC(C(=O)NCC1(C)CCCS1)NC(c1sncc1CC)=O N1(C(C(CC)O)=O)CCCC(CCNC(c2cc(C)n(C(C)C)c2)=O)C1 C1(C(N(CCNC(c2csc(C)c2C)=O)CC)=O)Cc2cc(C)c(C)cc2O1 c1(OCC)nc(N2CCC(N(C(=O)CN3CCNC(=O)C3)C)CC2)cc(C)n1 N1(C(C2(CC)CCC2)=O)CC2(C(=O)NC(c3cncnc3)C)CCC1CC2 C(=O)(CC(C)(C)N(C)C(c1ccc(CO)cc1)=O)NCC(C)N(CC)CC c1(C(=O)NC2CC(NC(c3cn[nH]c3)=O)C2)cc(C2CCCCC2)on1 Cc1nc(=NCC2CC(C)N(C(=O)C(C)SC3CCCCO3)C2)s[nH]1 c1(CC)nc(O)c(C(=O)NC2(CNC(c3cnnc(O)c3)=O)CCOC2)cc1C c1(C(=O)NC2CCN(C(C=C(CC)C)=O)C23CC3)ccc2c(ccn2C)c1 c1(C(CNC(c2c(CC)csc2)=O)NC(c2cnsc2)=O)cccc(C)c1 N1(C(CCC=CC)=O)CC(CNC(C2(CC)CC2(F)F)=O)C(C)C1 C1(C(=O)NC(C)Cn2cncn2)C2CCN(C(=O)Cc3ncccc3F)CC12 C1(NC(C)=O)CCCCNC1=O.c12cc(n(C)n1)C(=O)OC2.C1CO1 N1(C(c2c(C)noc2C(F)(F)F)=O)CC2CCC1CN2c1nc(Cl)ncc1Br C1(NC(Cc2cnc(C)o2)=O)CN(C(=O)CN(c2ccccc2)C)CC1C CN1CCN(C(=O)CCc2ccc(Cl)c(F)c2)CC1CNC(=O)Cn1ncnn1 C1(C(=O)NC2CCN(C(N)=O)C2)CCCCN1C(=O)C=CC1CCOCC1 N1(C(Cc2c(C)nn(CC(C)C)c2C)=O)CC(NC(=O)CC(C)O)C2(CCC2)C1 CC1CC(NC(=O)Cc2cc(C3CC3)nn2C)CN(C(=O)Cc2cnn(C)c2)C1 C(=O)(C(F)CC(C)(C)NC(C1CC2(CC(=O)C2)C1)=O)NCCCC1CC(C)C1 N1(C(CCSC)=O)CCN(CCN(C(=O)C(C)OC(C)=O)C)CC1 c1(C(N(CCCC(=O)NC(C#CC#C)(C)C)C)=O)cccc2c1CCC2 C(CNC(c1cc(C(N)=O)co1)=O)(C(=O)NOCCC(F)F)OC C1(C)(C(=O)NCC2N(C(c3cc(C)oc3C)=O)CCC2)CCNC(=O)C1 C1(C(=O)NC(CN(C(C=Cc2ccc(CC)o2)=O)C)(C)C)CC1C1CCCC1 C12(C(=O)OC)CN(Cc3cccc(CS(N)(=O)=O)c3)CC1CCCO2 c1(C2C(F)(F)C2CNCc2cncs2)cc2ccccc2nc1Cl c1(NCC(c2ccccc2)NC(C(C)CN(C)C)=O)nc2c(cc1C#N)CCC2 N1(c2cn(C)nc2)CCC(C(=O)NCC(F)CNC(=O)Cc2cccn2C)C1=O N1(CCN(C(=O)CC2CC=CC2)C)CCN(C(C2CSCC(=O)N2)=O)CC1 c1(C(N2C(CNC(C3CCCS3)=O)C=CC2)=O)cc2cc(F)c(F)cc2[nH]1 c1(COC(CN(C2CCSC2)C)=O)cc(C(F)(F)F)ccc1Br c1(C(=O)NCCCC(C)(C)NC(C(F)=C(C)C)=O)c(O)cc(=O)n2c1CCCC2 O=C1CCc2cc(C(N3CC(NC(=O)CSCc4ccc(F)cc4)C3)=O)ccc21 c12cnccc1CNC1CCN(C1)C2=O.C(=O)(CN(C1CCC1)C)NC C1(CC(C)C)(C(=O)NC(CNC(COC2(C#C)COC2)=O)C2CC2)CCNC1=O C1(C(=O)NCCCN(CC)CC)CCCC(C(N)=O)C1.C(=O)(C)NC(=O)CN(C)C C(CCC(C(=O)NCC(F)(F)F)c1ccccc1)NC(=O)OC CC(C#N)CN(C(C(=O)NCCCOCC1CC1)c1ccsn1)C1CC1 C12(NC(C(C)N3CCC3)=O)CCCN(C(=O)CCC(=O)c3ccncc3)CC1C2 N1(C(C2(NS(CC)(=O)=O)CC2)=O)CCS(=O)C(C)C1 C(=O)(C(C)C(O)CC)N1CCC(NC(Cc2nc(COC)sc2)=O)(CO)C1 C1(C(=O)NCC(C)NC(C2CC2c2ccccn2)=O)Cc2ccccc2N1 CCC(CC)(CC)C(=O)N1CCN(C(c2cn(C)cn2)=O)C(C2CCC2)C1 c1(C(=O)NCC#CCNC(Cc2n(C)nnc2)=O)ccncc1N C(=O)(CS(=O)(=O)C1CC1)NCC1OCC(C(N2CCC(CCC)C2)=O)C1 CC(CCC(C)(C)C)C(=O)N1CC(OCC(=O)OC(C)(C)C)C1 N1(Cc2cnc(C)s2)CCC2(CC1)CC(NC(=O)C(C)(C)O)CO2 Nc1sc2c(c1C(N1CC(C3(NC(C4CCCO4)=O)CC3)C1)=O)CCSC2 C1(C(=O)NCCc2cn(CC)nn2)(CNC(=O)CC(=O)OC)CC12CCC2 C1(C(=O)NC2(C)CC(C)C2)CN(C(C2(C)CCCOC2)=O)CC1C1CC1 C1(CN(C(C2CCCN2S(C)(=O)=O)=O)CC)CCCN1C(c1cc(C)c[nH]1)=O CCC(C(=O)NC1(C)CCN(C(=O)C(C)OCC2CC2)CC1)C(C)(F)F Cc1nc(C)c(C(=O)N(CCNC(=O)C(C)O)C2CC2)nc1C CN=c1[nH]c(=NCC2CCC3(CC3)C2)[nH]c(=NC2CC(Sc3cccc(F)c3)C2)[nH]1 CC1CN(C(C2SCCS2)=O)CC1NC(=O)CC12COC(C1)C2 c1(N(CCS(=O)(=O)NC)C)nc(N2CCC(C)(F)C2)c2cnn(C)c2n1 C(C(CC1CCCC1)C(=O)NCC(C)(O)C1(C)CC1)NC(C(C)(C)C1CCC1)=O C1(C(=O)NC2(CC=C)CCOC2)CC(=C)CCN1C(=O)C=C(C)C1CC1 C(CN=C(NCC1(N(C)C)CCCC1)NC(C)C)OC.c1(O)cncc(Cl)c1 c1(C(N2CC3CCCN(C(=O)C4=CCC4)C3C2)=O)cc(=O)n2nccc2[nH]1 Cn1[nH]c(=NC(=O)C(O)CCNC(C2CCCN2C=O)=O)cc1C(N)=O C=CCN(OC)C(=O)C1CCN(C(=O)CC2(C#N)CC2)C1(C)C C1(NC(C(C)OCCCC)=O)CCN(C(c2cncn2C)=O)CC(O)C1 c1(C(N2CC3C(N(C(=O)Cc4ccon4)C)C3C2)=O)cc([N+](=O)[O-])n[nH]1 C1(C(N)=O)CCC(C(=O)NCC(C2CC2)NC(C2(C3CCCCO3)CC2)=O)CC1 CC(CF)CC(=O)N1CCC(C)(NC(=O)Cc2ccc(F)cn2)C1 C1(C(=O)NC2(C(=O)NCC#C)CC2)C2CC3C(C2NC(C2(C#N)CC(=O)C2)=O)C13 Cc1ncc(C(N2CCC(N(C(=O)Cc3cnccc3Cl)C)C2)=O)n1C N1(C(CCCC)=O)CCC2(CC(C(=O)N(C)Cc3nccn3C)C2)C1 CCCC(C)CC(=O)NC1(C2CN(C(c3cc(OC)n[nH]3)=O)C2)CC1 N1(C(N=c2ccn(CCCC(=O)N(C)C)[nH]2)=O)CCC2(CCCC(C)(C)C2)C1 O=C(C1Cc2ccc(F)cc21)NCC1C2CN(Cc3ccns3)CC12 C1(COC)(COC(=O)OC(C)(C)C)COC1.C1(C)CNC(=O)N1 N1(C(CC(=C=C)C)=O)CC2CCCC(CNC(c3snc(O)c3Cl)=O)(C2)C1 Cc1ccc(C(F)C(=O)NCC(C)(O)CNC(c2cn(C3CC3)cn2)=O)cc1 C1(C(N(CC(C)(C)NC(C(F)=CCC)=O)C)=O)C2CC3CC(C2)CC1C3 CCCC(C)C(C(=O)NCCCOCC1CC1)N1CCCC2(CC1)CC2 C(=O)(CCC(C)C)N(C(C)(C)C)Cc1cn(Cc2nnc(C)o2)nn1 Cc1nc2sc1NC1CC(F)(C1)CNC(=O)NCC(=O)N2.C1(C2CC2)CCCO1 C12(CNC(=O)CCN3CCC3)CCC(NC(=O)CC3C=CCC3)(CC1)CC2 CC1(C)CC=C(C(=O)NCCC(O)CNC(=O)CN2CCC(O)CC2)CC1 N1(CC)CCOC(C(=O)N(C)CC2CN(C(=O)C(C)C(C)O)CCO2)C1 CC(=O)CC(C)(C)C(=O)N1CC2CC(NC(C3CCC(n4cccc4)CC3)=O)C2C1 C12(C(N3C(CNC(C(CCC)C(C)C)=O)CCC3)=O)CCC(OC)(CC1)CC2=O C(C(C(=O)NC(c1nncn1C)CO)NC(c1cc(CC)no1)=O)OCC C(=O)(C(=O)C(C)(C)C)N(C1CCCN(C(CC(C)c2ccncc2)=O)C1)C C1(C)(CC)CCN(C(=O)C(C2(O)CN(C(=O)CC3CCCNC3=O)C2)F)C1 c1(C(=O)NCC2N(C(CC(C)F)=O)CCOC2)c(F)cc(F)cc1F CCCCC(CC)C(=O)N1CCCCC(NC(=O)Cn2c(C)c(C)sc2=O)C1 CC1C(NC(c2ccncn2)=O)CC2CCC1N2C(c1c(F)ccc(F)c1N)=O C1(C(N(CCCCN(C(C(CC)SC)=O)C)C)=O)CC1C1CCCCC1 N1(C(C(CCOC)NC(c2cccc(C)c2)=O)=O)CCC2(CC1)CN(C)C2 Cc1cccnc1CNC(C(F)F)c1ccco1 N1(C(C(C)(C)C)=O)CCC2CC(CNC(C3CC34CCOC4)=O)CCC2C1 N1(CC(N2C(CCCC)CCC2)=O)CCC(Cn2cncn2)CC1 c1(C(=O)NC2CC(C(=O)Nc3cccc(F)c3O)C2)cc2ccccc2s1 N1(C(C(C)C)=O)CCCCC1C1CCCN(C(C2(C)CC2(F)Cl)=O)C1 C(CC(CC)C(=O)NCC1(NC(=O)C(C)OC2CCOC2)CCCC1)=CC c1(CC)ncncc1C(N1CC(O)CC1C(N1CCC1(C)C)=O)=O c1(C(=O)NCc2c(O)ccc(NCC)c2)nc2ccccc2s1 c1(C(=O)NC(CC)CNC(c2cc(O)nc(O)c2)=O)cccc2oc(C)nc12 C1(CC(=O)OC)CN(C(c2nnc(C)o2)C)CC(C)(C)O1 C1(NC(C(F)=CC)=O)CCC12CCN(C(=O)C(=Cc1ccco1)C)CC2 C(=O)(CCC(C)N(C)C)NC(c1nc(C(=O)NCCCOCCO)co1)C C1(NC(c2cn(CCC)nn2)=O)(CC)CCCN(C(=O)CCCc2cncs2)C1 c1(C(=O)NCC2C(NC(C3C(C=C)CC3)=O)CCC2)ccc(OC)cn1 N1(C(C=Cc2c(C)noc2C)=O)CC2CCC(C1)N2C(C1CN(CC(C)C)C1)=O Cc1nocc1C(N1CC(CCCCNC(=O)Cc2ccsn2)C1)=O N1(C(C(n2cc(Br)cn2)C)=O)CC2C(C(N3CC(F)C3)=O)C2C1 Cc1n[nH]c(C)c1C(C)C(=O)NCC1(C)CC(NC(=O)CS(N)(=O)=O)C1 N1(C(C(C)OCC=C)=O)CCCC(CC)(NC(c2cc(C)cc(N)c2)=O)C1 C1(C(=O)NC2CN(C(c3c(CCC)n[nH]c3)=O)CC23CC3)CCc2nc[nH]c2C1 c1(C(CC)N(C(c2cocc2Br)C(=O)NC2CCCOC2)C)c(C)nn(C)c1C C1(C(=O)NC(CCCC)CNC(=O)C(CN(C)C)N(C)C)CCS(=O)(=O)CC1 CC1CN(C(c2c(C3CC3)cnn2C)=O)CCCN1C(=O)Cc1ccn(C)n1 Cc1ccc2oc(=NCC3CN(C(c4cc(C(C)(C)C)no4)=O)CC3C)[nH]c2c1 c1(CNC(C(C(C)OC)O)=O)n[nH]c2c1CN(C(=O)CSC(C)C)CC2 N1(C(C2CCNC2=O)C(=O)NCCCSC)CCC2CC(c3ccccc3)C2C1 C1(N(C(c2cc(C)nn2CC)C(=O)NC)CC)CCC(F)(F)C1 C(C(CC(=O)N1CC2CC1C2NC(c1nccc2[nH]ccc12)=O)C(F)F)N(C)C N1(Cc2cn(CC=C)nn2)CCCN(C(C2(O)CCOC2)=O)CC1 N1(C(=O)NCCCl)CCC2CN(C(c3c(Cl)cc(Cl)cc3Cl)=O)CC2C1 N1(C(COc2ccc(COC(Cn3ccc(C)n3)=O)cc2)=O)C(C)CCCC1C C1(C(=O)NC(CC=C)(C)C)CC2CC1CN(C(=O)C(O)CSC)C2 CCC(CC)(CC(=O)OC)C(=O)N1CC(NC(c2ccc3nn[nH]c3c2)=O)C1 C(=O)(CS(=O)(=O)CC1CCCO1)OCC1(OC(C)C)CCOCC1 C1(C(=O)NCC(C2CCN(C(CC(=O)OC)=O)CC2)(C)O)CC2COCC(C1)C2 C(=O)(C(F)(F)C(C)O)NCC1CCN(C(C(C)c2ncco2)=O)CC1 N1(C(CCC(CC)NC(c2c(C)cccc2O)=O)=O)CCn2ncc(O)c2C1 c1(C(=O)NC(C(=O)OC)Cc2ccccc2Br)ccc2c(c1Cl)OCO2 c1(C(c2n(CC)nnn2)NCCC(=O)OCC)ccnc(NC2CC2)c1 C1(NC(C(C)(C)OC(C)C)=O)CN(C(c2ccc(C3CC3)s2)=O)C2(CCCC2)C1 c1(C(N)=O)ccc(C(=O)NC2CCC2NC(C2(n3cnnn3)CC2)=O)nc1 C(CC(CO)C(C)C)NC(C1(SC)CN(C(C2OCCC2(C)C)=O)C1)=O c1(CNC(C2CC(CF)C2)=O)ncc(Cn2cc(C(=O)O)nn2)o1 c1(CC(=O)NC2CCC(NC(C)=O)CC2)ccc(C)cc1Br CC1CN(C(c2cc3n(n2)CCC3)=O)CCC1NC(c1c[nH]nc1C(C)(C)C)=O N1(C(C(c2ccccc2)NC(c2c(N)nccn2)=O)=O)CC2C=CC1CC2 C(CCCCNC(=O)C(=O)NC(c1cc[nH]n1)C1CC1)OCCOC Cc1ccccc1CCC(=O)NCCCCCNC(=O)C(C)(C)CO c1(C(N2CC3C(C(=O)NCc4cn(CC)nc4)(C3)C2)=O)ccc2c(c1)NCCO2 c1(CCC)ccccc1NC(C1CC(F)CN1C(c1cccs1)=O)=O c1(CNC(C2CC(NC(C3N(C(C)=O)CSC3)=O)C2)=O)cc(Cl)c(Cl)cc1C C1(NC(CN(C(COC)=O)C)=O)CN(C(c2ccnc(CO)c2)=O)CCC1F C1(NC(CN(CCC#C)C)=O)COC2(CCCN(C(=O)C(=O)N=S(C)(C)=O)C2)C1 C1(C(=O)NCC2CN(C(C3OCCN(C)C3)=O)C2)CCCC12CCOCC2 Cc1cc(F)ccc1C(N1CC(O)CCC1C(=O)N(C(CF)CF)C)=O Cc1ccc2cc(C(=O)NC3CCC(NC(c4[nH]nnc4C)=O)C3)ccc2c1 c1(CC(C(=O)NCC2CN(C(c3ccn(C(C)C)n3)=O)C2)C)ccc(O)cc1 C1(CC)CN(C(=O)CCC(C)OC)CCC1NC(c1cc(C(C)C)n(C)n1)=O c1(C(=O)NC2CCC(CNC(=O)CCc3ncc[nH]3)C2)c[nH]c2cc(O)ccc12 CC1COCC(C(=O)NCC2CCN(C(=O)Cc3cnn(C(F)F)c3)CC2)O1 O(N(C)C(=O)CNC(=O)C(C)NC(=O)CC1CC(=O)C1)CC C(=O)(C(C(C)OC)N(C)C)N1CC(CCCCNC(c2c(CC)csc2)=O)C1 Cc1cc(C(N2CCCC2CNC(C2C3(CC3)C23CC3)=O)=O)cnc1C(F)(F)F C(CC(C(=O)Nc1ccc(SC)cc1)NC(c1occc1C)=O)OC c1(C(N(C2(CCN=[N+]=[N-])CC2)CCO)=O)cc2c(nc1Cl)CCS(=O)(=O)C2 N1(C(c2cc(C)cc(Cl)c2)=O)CC(NC(=O)CC2CC3(CC3)CO2)CC12CCC2 N1(Cc2n(C)ncc2)CC(NC(c2ccc(F)c(C3CC3)c2)=O)C(C)(C)C1 N1(C(CCC2CCC(C)O2)=O)CCC(C)(CNC(c2cc(O)ccc2O)=O)CC1 C1(CNC(c2c(CC)c[nH]c2)=O)CC(F)(F)CN1C(c1ccc(C)c(Cl)c1)=O c1(C(=O)NC2C=CC(CNC(C(C(C)(C)C)O)=O)C2)ccc2cccnc2n1 N1(C(C(CO)N(C)C)=O)CCC(C2CN(C(=O)COc3cccc(F)c3)C2)CC1 C1(NC(CN(c2ccncc2)C)=O)CCC(NC(=O)C(O)C2CCC2)C1 N1(C(C2(NC(CCCOC(C)C)=O)CCCC2)=O)CCc2n[nH]cc2C1 c1(CC)cnccc1C(=O)NC(C)C(CO)NC(=O)C(C)Oc1cccc(F)c1 C1(C(=O)OC)CC2(CCC1NC(c1cc(C(N)=O)ccc1C)=O)CC2 c1(C(=O)NC(C(=O)OCC)C2CC2)cn(CCNC(C2(CO)CC2)=O)cn1 C1(NC(c2cccc(OC)c2)=O)CC1C1CCCN(C(=O)C(C2CC2)C2CC2)C1 C1(NC(C=CC(C)C)=O)CCC(C(=O)NC(c2ccccc2F)C2CC2)OC1 c1(C(N2C(CNC(=O)Cn3cc(Br)cn3)C=CC2)=O)cc2cc(F)ccc2s1 N1(C(c2c(OC)cccc2)=O)CCN(C(=O)Cn2cnnc2O)CC1CC(F)F c1(C(=O)NCC(N2CC(C(C)CNC(c3nocc3C)=O)C2)=O)ncccc1O N1(C(CCC(C)OC)=O)CCN(C(c2ncn(C)n2)=O)C(c2cn[nH]c2)C1 C(c1cc[nH]n1)=CC(=O)NCCC1CN(C(CC2(C)CC2F)=O)C1 C1(OC)(CNC(c2nc(Cl)cs2)=O)CCN(C(C2CC3CCC2O3)=O)C1 c1(C(N(C2CN(C(C3C4CCCCC34)=O)CC2(C)C)C)=O)[nH]cc2c1CCCC2 Cn1ncc2c(N3CC4CCC3C4)nc(=NC3c4c(F)cccc4CC3C)[nH]c12 CC(C)C(F)C(=O)N1CCC(CNC(c2ccccn2)=O)C1 c1(C(N2CC=CC(NC(C(c3ccccc3)OC)=O)C2)=O)cc(F)ccc1C C(CC(CC)C(=O)N1CC(C)(NC(=O)CCn2cccc2)C1)=CC C1(C(=O)NCC(C)CNC(=O)CCCC2CCCC2)CN2CC3CC2(CO1)C3 c1(C(=O)NC2C(C)CN(C(=O)CCN3CCC3)C2)ccc2c(c1)C(=O)NC2 N1(C(c2csc(NC=O)n2)=O)CC(O)C(O)C1CNC(CC(C)NC(N)=O)=O c1(-c2c(C(=O)NCc3cccc(N)c3)ccnc2)c(F)cc(F)cc1F c1(CNC(C2N(C(COCCOCC#C)=O)CC2)=O)ccc2c(n1)NCC2 C(C(=O)N(CC(O)CNC(=O)CCOc1ccc(CC)cc1)C)(C(C)C)SCC N1(C(C2CCN(C(C3CC(C)C(=O)CC3)=O)CC2)=O)CCN2CCCC2C1 CC1=NOC2(C1)CC(C(=O)Nc1c(C)nc(O)nc1S)C2.c12ccc(cc1)CO2 c1(OC)ccc(C(=O)NC(C2CCCC2)CNC(c2coc(Cl)n2)=O)cc1 C1(NC(C2CCOC2(C)C)=O)C=CCC(C(N(C2CCC3(CC3)C2)C)=O)C1 C1(CCOC)(NC(=O)C(C)Nc2cnn(C3CC3(F)F)c2)CCOC1 C1(NC(C=C(CC)C)=O)(CNC(=O)CC2CS(=O)(=O)C2)CC2CCC1CC2 N1(C(COC2(C)CN(C(=O)Cc3ccco3)C2)=O)CC2CCC(O)CC2C1 C12(C(N3CC(N(C(=O)Cn4cnc(C(N)=O)n4)C)C3)=O)CCC(C1)OC2 c1(C(=O)NCCCN(C(C2CCCCO2)=O)CC)cc2cc(Cl)cnc2[nH]1 c1(C(=O)NC2CCN(Cc3c(CC)cccc3)C(C)C2)cnc2ccccc2n1 c1(CC)c[nH]nc1C(=O)NCC(C)C(=O)NCc1cc(O)ns1 CC1(C)C(NC(=O)C(O)Cc2ccc(F)cc2)CCN1C(=O)C=Cc1ccc[nH]1 c1(CC)ccncc1NC(=O)C(CCN(C)C)NC(=O)CCOCCOC c1(Cc2onc(C(C3CC=CCC3)OC)n2)c(Cl)cccc1Cl c1(CC)ccccc1C(c1nnnn1C)NCC1(c2ccccc2)CC(O)C1 C1(S(C)(=O)=O)(C(N(C(C)CNC(=O)C(N2CCOCC2)C)C)=O)CC1 C(=O)(C#CC(C)C)N1CCC(C(C(=O)NCc2snc(C)n2)C)C1 c1(C(N2CCC(F)(C(F)F)C2)=O)ccc(-c2cn(CCCCF)nn2)c(Cl)c1 N1(C(C2C(CC)N(C)CC2)=O)CCN(C(c2cccc(C3CC3)n2)=O)CCC1C c1(C(N(C)CC2N(C(c3n(C(C)C)ncc3)=O)CCC2)=O)ccc(Cl)nc1O N1(C(C2OCCN(C)C2)=O)CCC(C)(C)C1C(=O)Nc1ccc(OCF)cc1 N1(C(Cc2nc(CC)sc2)=O)CCC(O)C(NC(=O)CC2(C)CCS(=O)(=O)N2)C1 C1(NC(C(C)OCC=C)=O)(CNC(C2CC=C(C)CC2)=O)CCOCC1 Cc1ccc(F)c(C(=O)NC2CC(NC(=O)C3=CCCC3C)CC2O)c1 C1(CCNC(c2c(C)scc2)=O)CC(F)(F)CN1C(=O)C=Cc1cncc(O)c1 CN1C(=O)CC(NC(C2CC(O)CN2C(=O)CCc2nncn2C)=O)C1=O c1(OC)ccc2c(C(N3CCC(Oc4ccccn4)C3)C(=O)NC3CC3)n[nH]c2c1 c1(C(=O)NC2CCCN(C(c3cc(C)c(F)cc3)=O)C2C)ccn2nccc2n1 S(=O)(=O)(c1c[nH]c2cccc(OC)c12)N(CC(=C)C)CC12CC(CCO1)C2 N1(C(Cc2nc(C)oc2)=O)CCCC2C1CCCN2C(C1CC(=C2CC2)C1)=O Cc1cc(C(=O)NNC(=O)c2ccc(-c3ccccc3)s2)nc(Br)c1 N1(C(C(=O)OCC)=O)CCC(NC(=O)C=C(C)c2ccc(OC)cc2)C(C)(C)C1 c1(CC(C)NC(=O)Nc2c(COC)cccc2)ccc(Br)cc1F CC(C)C(C)CC(=O)N1CC2CC(NC(=O)C(F)(F)c3cncs3)C1C2 S(=O)(=O)(CCCN=c1[nH]c(=NCC(c2ccccc2)N(C)C)[nH]c2cc[nH]c12)NC N1(C(C2CC(NS(=O)(=O)Cc3ccc(Cl)c(Cl)c3)C2)=O)CCn2cnnc2C1 CCC(F)(F)CC(=O)N1CCC2(NC(c3cn(C)cc3C)=O)CC2C1 C1(C(C)NC(C2(C)CC(=C)C2)=O)CN(C(=O)C2=CCCO2)CCO1 C1(NC(c2cccc(CC=C)c2)=O)CCC(C)N(C(=O)CSCCOC)C1 N1(Cc2[nH]c(=N)sc2C(F)(F)F)CCCC(NC(=O)Nc2ccccc2)CC1 c1(C(C)C)[nH]ccc1C(=O)NCC1CCCC1NC(=O)C(O)C1CCCC1 c1(-c2nc(-c3scc(C)n3)nn2C2CC3CCC2C3)csc2cc(Cl)cnc12 N1(C(C2C(OC)C2)=O)CC23CCCC2(C1)CN(C(c1ccc(CC(C)C)s1)=O)C3 c1(C(N(C)CC2N(C(c3c(COC)nn[nH]3)=O)CCC2)=O)c(C(C)C)cnn1C c1(C(N2C(C(C)NC(CC(=C=C)C)=O)CCC2)=O)cc(C)c(F)cc1N C1(NC(Cc2n(C)nnc2)=O)(CO)CCN(C(c2ccc(C#N)cc2)=O)CC1 c1(C(=O)NCC(C2CC2)NC(CSCCOC)=O)c(C(C)C)cccc1F c1(CC)noc(C(=O)NC(c2ccc(C)cc2)CNC(C2CCCO2)=O)c1C [N-]=[N+]=Nc1ccccc1C(=O)NCC1(NC(=O)C(F)=CC2CC2)CCCCCC1 Fc1ccccc1SCc1nc(-c2cc[nH]n2)nn1C1CC1 N1(C(C)C(=O)OCc2nn(C)cc2Br)C(=O)C2CCCCC2C1=O C#Cc1cccc(CC(=O)NCC2CC(NC(C3(CC)CCCO3)=O)CCO2)c1 c1(CN2C(CC(=O)Nc3c(OC)nnc(Cl)c3)CCC2)c[nH]c2cccnc12 CC(C)C(O)C(C)(C)C(=O)NCC1CCN(C(c2ccc3nc[nH]c3c2)=O)CC1 CC1(NC(c2ccc(C3CCC3)nc2)=O)CCN(C(c2csc(Cl)n2)=O)C1 N1(C(C=C)=O)CCN(CCCC2CCN(C(c3cnc(C(C)C)s3)=O)CC2)CC1 C1(CC(=O)NC2C(C=C)CN(C(C3CC(F)(F)C3)=O)C2)CC2(CCCC2)CO1 CS(=O)(=O)CCCCCCCC(=O)N1CC2CC1CN(C(=O)C1=CCSC1)C2 Cc1cccc(CC(N2CCCCC(N(C)C(c3ccnnc3O)=O)C2)=O)c1C n12cc(nn1)C(=O)N1CC2C1.C(=O)(CC(=O)NC1CC1)NCC1C(=C)C1 C1(C(=O)NCCOCCNC(C2CCCCCCC2)=O)CCCCC12CC2 N1(C(C(c2cccnc2)NC(c2n(CCC)ncc2)=O)=O)CC2(CC2)CC1C N1(c2snc(C(=O)OC)n2)CCCC(C)(C(=O)NC2COCC2O)C1 N1(C(C2(C)N(C)CC(OC)C2)=O)CCC2(CCCCC2NC(=O)CSC)CC1 C(C(CCNC(c1cc(C)on1)c1nnnn1-c1ccccc1)C(C)C)OC c1(CNC2CN(C(c3cnc(NC(C)=O)o3)=O)CC2F)ccc2c(C)c[nH]c2c1 Cc1cc(C(N2CC(NC(c3cnc(S)nc3)=O)CC2C)=O)ccn1 Cc1c[nH]c(C(N2CCC(CCCNC(C3CC3C)=O)CC2)=O)cc1=O C12(NC(c3ncn(C)c3)=O)CCCC1(F)CN(C(C1CC1(Cl)Cl)=O)C2 c1(C(=O)NC2(CC=C)CN(C(=O)Cc3cscn3)C2)cnn2cccc(C)c12 N1(C(c2c(C)cccc2C)=O)CC2CC(NC(=O)CN3CCCS3(=O)=O)CC1C2 C#Cc1ccc(C(=O)N(CC(N2CCCC3(CC3)C2)=O)C)c(C)c1 C(C(C)(C)C(=O)NC1CC(C)(C(=O)NC2CCN(C(C)C)C2)C1)NC(C)=O c1(C(=O)NC2CC(C)(CNC(C(CC)n3ccnc3)=O)C2)cc(C)ncc1C N1(C(C(CC#C)(C)C)=O)CC2CCCC(CNC(=O)C(CC)SC)C2C1 c1(C(=O)NC2CC(NC(c3ccc(C)c(C)c3)=O)C2)cc2c(cc1O)CCC2 C1(NC(C(C)NC(=O)NC)=O)CCN(C(=O)C(c2ccc(F)cc2C)O)CC1C c1(C(=O)NC2CN(C(CC3C(C)(C)C3)=O)CC(F)C2)ccnc2[nH]cnc12 c1(CN2C(C)(C(=O)Nc3cccc(CCO)c3)CC2)cc(O)cc(Br)c1 c1(C(N2CC3CC2CN3C(=O)C(F)(F)F)=O)cc2cccnc2nc1O C1(N(C(=O)CNC(=O)NC2CC2)C)CCN(C(=O)CC2CNC(=O)O2)C1 CCC(C)CCC(=O)N1CC2(CC2)CC1CNC(=O)CCc1cccc(F)c1 N1(C(CCCN(CCC)CCC)=O)CC(N(C)C)C(NC(=O)C(C)(C)CSC)C1 CC(O)(CNC(=O)CCNc1ccccc1)CNC(=O)CCN1CCOC1=O N1(C(c2n(C)nc(O)c2)=O)CCCC(C2(NC(=O)CCCS(C)(=O)=O)CC2)C1 C1(C(N2CC(C)(NC(C(C)OC3CCCC3)=O)C2)=O)CCC=CCCC1 C12(C(N(C3CC(NC(C4CC5C=CC4O5)=O)C3)C)=O)CCCN1CCC2 C12(CNC(c3c(C)ccnn3)=O)CCCCC1N(C(c1cncnc1C)=O)CC2 c1(C(=O)NC2CC(CNC(C(c3ccnn3C)C)=O)C2)ccnc(C(C)(F)F)c1 c1(CN(C)Cc2c(CC)cccc2)ccc(S(=O)(=O)N(C)C)cc1 c1(CC)cc(C(=O)NCCC2(CNC(c3cc[nH]n3)=O)CC2)nn1C CC1(CC(N2CCC(NC(C3CC3C#N)=O)C2)=O)OCCO1 c1(C(N(C(C)CNC(c2cnn(CC)c2)=O)CC)=O)c[nH]c2ccc(Cl)cc12 C#Cc1cn(C)nc1C(=O)NCC1(COC)CN(C(C2(C)CC3C=CC2C3)=O)C1 c1(OC)cccc(CC(N2CC(N3CCN(C(c4nccs4)=O)CC3)C2)=O)n1 Cc1cc(C(N2CCC(F)C(NC(c3cc(Cl)ccc3C)=O)C2)=O)c(C)cc1Br c1(C(N2CCC3(CN(C(CC(CC)C)=O)C3)C2)=O)ccc([N+](=O)[O-])c(N)n1 O=C(CS(=O)(=O)C1CCCC1)NC1C2CC(O)C1N(C(C1(CO)CCCO1)=O)C2 Cc1cccc(CC(C)(O)C(C)NC(=O)N(C)CCc2ncon2)c1 N1(C(c2c(C)cc(C)s2)=O)CC(N(C(=O)Cc2cn(C)nn2)C)C(C)(C)C1 c1(-c2ccc(C(=O)Nc3c(C(=O)OCC)cc(C)s3)nn2)cccc2ncoc12 c1(-c2nn(C(CC)C)c(CN3CC4CC4C3)n2)ccc2ccccc2n1 C1(NC(N2CCC(C(=O)N3CCCc4nccn43)CC2)=O)C2Cc3cc(F)ccc3C12 N1(C(c2c(C)nc(COCC)s2)=O)CCCC(F)(CNC(C2(C(N)=O)CC2)=O)C1 c1(C(=O)Nc2n(CC(C)C)ncc2)ccccc1C1=CCOCC1 c1(N2CCC(NC(c3cnncc3O)=O)C2)cc2nncn2cn1 C1(NC(CSCCOC)=O)(CNC(=O)C(F)(F)C2(O)CCC2)CCOCC1 CC1(C)CC2(CC2C(=O)NC2CCCCC2NC(c2cc(C3CCC3)on2)=O)C1 N1(C(c2c(CC)nn[nH]2)=O)CCC(O)(CCNC(c2ccc(C3CC3)nc2)=O)C1 C1(C(N2CCCN(C(C3C(C)C3)=O)CC2)=O)CCc2nc(C(C)C)[nH]c2C1 C(=O)(C(CN=[N+]=[N-])NC(c1cc(CCC)on1)=O)N(C(C=C)C)C C(=O)(C(O)C(C)(C)C)NC(CC)(C)CNC(c1cccc(C2CC2)c1)=O C(=O)(CCCCOC)NC.C1(C)C(=O)N1CCCc1nccs1 Cc1ccccc1-c1cccc(C(=O)NCC2C3CN(C(=O)CC(C)O)CC23)c1 C1(NC(C2(CO)CCN(C(=O)C(O)CN3CCCC3)C2)=O)CC2(C1)CC(O)C2 N1(C(CC(CC)C2CCC2)=O)CCC2CN(C(C3(CCOC)CC3)=O)CCC12 N1(C(C2ON=C(C)C2)=O)CCN(C(=O)CC(C)(C)c2ccc(F)cc2)C2CCC12 C1(C(=O)NCC2(CNC(C(C(C)C)C#N)=O)CCCC2)CCC2(CCOCC2)C1 c1(Nc2cc(OC(C)C)ncn2)cccc2nc(O)n(C)c12 C=CCC(C)(C)C(=O)N(C)CC1CCCN(C(c2cc(C(C)C)oc2C)=O)C1 N1(C(C2CSC2)=O)CCCC2(C1)CN(C(C1CC13CC(O)C3)=O)CCO2 c1(C(=O)Nc2cc(F)cc(Cl)c2)ccc2ncc(C3=CCNCC3)n2c1 C(=O)(C(O)CC(C)(C)C)NC(CC)CCC(=O)N1CCCNC(=O)C1 O=S(=O)(c1cccc(Cl)c1)NCC1CCC2(CNC2)O1 CCCCC(C)C(=O)N(CCCNC(c1[nH]c(C)nc1CC)=O)CC c1(-n2cc(-c3c(C)noc3)nn2)cnc(C(=O)NC2CC2)nc1C(F)(F)F c1(C(N2C(CN(C(C(CC)O)=O)C)CCC2)=O)ccn2ccnc2c1 N1(C(C(CC)N(C)C)=O)CCC(C)(C)C(C(=O)NC(c2ccccn2)CO)C1 c1(C(=O)NCC(CNC(C2(C)CCC2)=O)OC)sc(C)nc1C(C)(C)C C(=O)(CCCCNC(N)=O)N(C1CCN(C(=O)C(C)C(F)F)CC1)CC c1(C(=O)Nc2ccnc(-n3cc(C4CC=CCC4)nn3)c2)cnc2ncccn12 c1(SCc2cc(OC)ncn2)cc(O)c(Br)cc1[N+](=O)[O-] C1(F)(C(N2CCC(CC)C2)=O)CCN(C(C2(Cl)CC2(F)F)=O)C1 C1(NC(c2cc(C)no2)=O)CCC2CC1CN2C(=O)CSCC(F)(F)F c1(C(=O)NCCC2CCCN(C(c3nncs3)=O)C2)ccc2ccoc2c1 C1(CNC(CC(COC)C)=O)CC2COCC2N1C(c1cc(=N)[nH]c(=N)[nH]1)=O c1(N2CC(C)S(=O)C(C)C2)c([N+](=O)[O-])cnc2ccsc12 CC1=CCCN(N(CC2CCC2)Cc2ccccc2Cl)C1 c1(C(N2CCCC(N(C(=O)CCC#N)C)C2)=O)ncc(P(C)(C)=O)cn1 C(=O)(C(F)(F)CC1CCCCC1)NCC1CN(C(CC(=O)NCC#C)=O)C1 CC(CCC(=O)OC(C)(C)C)NC(=O)Nc1ccc(Cc2nn[nH]n2)cc1 N1(C(CN(C)CC)=O)CC2(C)CN(C(c3ccnc(Cl)c3Cl)=O)CC2(C)C1 c1(OC)ccc(F)cc1CN1CCC(O)CC1c1ccccc1 c1(N(C(C(CNC(CC(CC)C2CCC2)=O)N(C)C)=O)C)cccc(C)c1C CC(C)(C(=O)NCC1CNC(=O)C1)C1=CCN(C(=O)CCCN=[N+]=[N-])C1 Cc1nc(N2CCCC(C(=O)Nc3cc(C)c(Br)c(F)c3)C2)c2c[nH]nc2n1 N1(c2cc3nnc(C)n3cn2)CCCC12CCN(C(=O)COC(F)F)CC2 C1(C(=O)NCC(CSC)OC)CCC2CCC1N2C(=O)C(C)(C)CC#N CC(C(=O)NC1(C)CCN(C(=O)CONC(=O)OC(C)(C)C)C1)C(F)(F)C(F)F c1(NC(C2CC3(CC3)CN2C(=O)Cc2ccc(O)c(O)c2)=O)cnc(Cl)cc1I c1(C(CN(C2CCN(C(=O)C(=O)NC3CC3)CC2)C)=O)csc2c1CCCC2 C(=O)(C(CCC1OCCO1)N1CCSCC1Cc1ccccc1)NC(C)C N1(C(c2c(OC)nccc2)=O)CC2CC(C1)N(C(=O)CS(=O)C(F)(F)F)C2 N1(C(C=COCC)=O)CCCCC1C(C)NC(c1c(Cl)csc1Cl)=O N1(C(CC2(C=C)CC2)=O)CCN(C(=O)C=Cc2ccco2)C(C)CC1C N1(C(Cc2c(C)nn(C)c2)=O)CCN(C(C2CCOC2C)=O)C(c2cn[nH]c2)C1 C1(C(=O)NCc2ccc(OC)o2)C2CCN(C(C3(CC4CC4)CC3)=O)CC12 CCCC(C(C)(C)C)NC(=O)CCN(C(C1CCCCC1O)=O)C(C)C N1(C(C2(CCSC)SCCCS2)=O)CCCN(C(=O)CC23CCCC2C3)CC1 c1(C(=O)NCC2N(C(C(C=C)O)=O)C3CCC2C3)cc(N)c(O)c(F)c1 c1(C(=O)NC2C(NC(c3cn(CC(F)(F)F)nn3)=O)C2)c[nH]cc(Cl)c1=O c1(SC)ncc(C(=O)NC2CCC(NC(=O)C(C)Cn3ccnc3)CC2)c(O)n1 c1(C(N(CCC)CCNC(C2CCC(C)O2)=O)=O)cc(Cl)nn1-c1ncccc1Cl C1(CN(C(c2ccc(C(F)(F)F)s2)C(=O)NCc2ccco2)C)CCCOC1 CC1(C2CCC2)CN(C(C2(NC(C3CC=CCO3)=O)CCSC2)=O)C1 c1(C2C(C(=O)OCC3CCOCC3)C2)ccc([N+](=O)[O-])cc1 CC#CCC(C(=O)NCC1C2CCC1CC2)NC(=O)COCCOC C#CCC(C(=O)NCc1ncccc1COC)NC(=O)Cn1c(O)nnc1O c1(CNC(c2cc(CNC(C(C)NC=O)=O)sc2)=O)ccc(O)cc1 CCC(CC)CCCN(C(=O)CC1CN(C(=O)COC(C)(C)C)CC1OC)C CCC(O)C(F)(F)C(=O)NCCCCN(CCCNC(=O)CCCCCCSC)C CC1=C(C(=O)NC2CC2CNC(C2(C(C)(C)C)CCC2)=O)CCO1 c1(C(CCC)NC(=O)CC2CCCS2)ccc(-c2cn(CC(=O)OC)nn2)cc1 c1(C(=O)NC(C2OCCN(C(C3(C)C(CC)CCC3)=O)C2)C)cc(C)nnc1O C1(NC(=O)NCc2ccc(-c3nc(C)on3)cc2)CCCC1C1CC1 N12CCC(CC1C)NC2=O.C1(C(=O)NCC2(CC(C)C)CC2)COC(C(C)C)C1 C(=O)(C1=CCCCCC1)NCCC1CC(NC(C2(C)CCC(=O)N2)=O)C1 C1(NC(C2C(C(=O)OC)CC2)=O)CC12CC(NC(C1(C)CC1)=O)C2 N1(C(C2CC(CC)C2)=O)CCCCC1CN(C(=O)C(C1CCOCC1)F)C CCCCC(C)C(=O)NC1CCC12CN(C(c1cc(-c3cn(C)nn3)on1)=O)C2 c1(NCCNC(C(=O)N(CC(=C)C)C)=O)cccc(C(=O)OC)c1 N1(C(C(CC)NC(C)=O)=O)CCOC(CNC(c2cnoc2CCC(C)C)=O)C1 C(=O)(C1CCCc2cccnc21)NC1(C)CC(NC(c2cc(C#N)ccn2)=O)C1 Cc1ccc(OC(F)F)cc1NC(=O)Cc1nc(Br)sc1C c1(C(N(CC(C)O)CCNC(c2c(C)cn(C)c2)=O)=O)cnc2ncc(Cl)cn12 CCCCC(CCC)NCc1cn(-c2ccc(C)cc2C)nn1 C=C1CC(C(=O)NC2CC2)(CNC(=O)C(=O)NCc2nc(C)cs2)C1 c1(OCC)ccccc1N1CCN(C(C(=O)NC2CCOC2)C2CCC2)CC1 CC(C)CC1C(=O)N1.N1(C(C(=O)OC(C)(C)C)=O)CCC(CCS(C)(=O)=O)CC1 C(N=c1nc(N2CCC3(CC2)CC3(F)F)c2c([nH]1)COC2)c1c(Cl)cccc1 C1(CNC(CC2CC(OC)C2)=O)CC2CCC(C1)N2C(=O)COC1CC=CC1 CC(CNC(c1[nH]cc2c1CCC2)=O)CC(=O)N1OC2C=CC1CC2 c1(C(=O)NC(CC)CNC(=O)C(F)(F)C(C)O)ccc(C)c2ccccc12 CCC(C)(C)C(O)C(=O)NC1(CF)CCN(C(=O)Cc2ccc(C(=O)OC)cc2)C1 c1(C(=O)NC2C(C)(NC(C3C(=C)C3)=O)CCC2)cccc2c[nH]nc12 n1(C(c2cc(C(N)=O)no2)C)c(-c2cc(C)ccc2C)csc1=Nc1ccc(Cl)cc1 C1(C(N2CCC(CCOC)(NC(=O)C3=C(C)OCC3)C2)=O)CCCC12OCCO2 C1(CCC(=O)NCCCNC(=O)CNC(c2ccccc2)=O)NC(=O)NC1=O c1(CNC(C)(C)CN2CCSCC2)cc(F)cc(Br)c1 N1(C(C(C(C)C)S)=O)CCC12CCN(C(=O)C=Cc1cccnc1)CC2 c1(-c2n(CCOCC=C)c(N3CCCOC(C)C3)nn2)csc2cccc(F)c12 CC(C)C(O)C(C)C(=O)NC1CCN(C(c2ccnc(C(F)(F)F)c2N)=O)CC1 CN1CC(C(=O)NCC2(C)CCCN2C(=O)Cc2cccc(Cl)c2)NC1=O N#CC1(C(=O)NN2CCC(c3ccccc3)CC2)CCCO1.C12CN(C1)C(=O)N2 C(C)(C(=O)NC(C(=O)NC1CC=CC1)C1(O)CCC1)OCC#C c1(C(=O)NCC(C)(C)OCC(N2CCC2C2CCCCO2)=O)coc(CO)c1 c1(CC)cnc(C(C(=O)NC2CCOCC2)N(CC(=O)OC)C)o1 c1(C(C(=O)NC2(CF)CCN(C(c3ccc[nH]3)=O)C2)O)ccc(F)c(Br)c1 c1(OC)cc(C)cc(C(N2CCC(NC(=O)CN(C)S(N)(=O)=O)C(C)C2)=O)c1C c1(COC)cccc(C(=O)NCC2CC(OC)CN2C(=O)CCCC#N)c1 C(=O)(C(C)(C)CCCC(=O)N1CC(NC(=O)CCc2nnc(C(F)F)o2)C1)OC c1(C(=O)NCC(C)N(C(C(C)=C2CC2)=O)C)nc(C)n2c1CCCC2 C(C1CCCn2cc(C)nc21)NC(c1cccc(SCCC)c1)=O c1(C(c2nnnn2C2CC2)NC(c2nc(C(C)(C)C)cs2)C)ncccc1Cl C1(C(=O)NCC2(C)CCCN2C(=O)CC2CCCC2)COC2COCC12 C1(NC(c2ccn(CCOC)n2)=O)CCC(NC(=O)CC2CCCC(=O)N2)CC1 C1(CNC(c2cnc(OCC(F)F)cn2)=O)CCCN(C(C2(F)CCCC2)=O)C1 CCCC(C)CC(=O)NCC1CCC(NC(=O)C=CCN2CCOCC2)C1 Cc1cc(C(=O)NC2CCC(C(=O)NC3CCSCC3)CC2)nc(C)c1 N1(C(c2ccn(C)n2)=O)CCN2CCN(C(=O)Cc3cccc(Cl)n3)CC2C1 c1(NC(c2ccc(C#C)cc2)c2nnnn2CCCC)ccccc1C(=C)C Cc1sc(NC(N2CCC(C(=O)N(C)C(C)C)CC2)=O)nc1C(C)C N1(C(c2cc(OC)n[nH]2)=O)CCCC(O)(CN(C(=O)Cc2cc[nH]n2)C)C1 C1(NC(c2c(Br)c(CC)n(C)n2)=O)CCN(Cc2cc(B(O)O)co2)CC1(C)C c1(C(N(CCNC(c2cc(OC)ns2)=O)C2CC2)=O)cccc(C2CC2)c1Cl Cn1nc(C(=O)NCC2CC(NC(=O)C(O)C3CC3)C2)cc1-c1ccc(Cl)cc1 CCC(C)(COC)C(=O)NCCn1cnc(C(=O)NC(C)CC(C)(C)C)c1 c1(SCC)cc(C(=O)NCCOC2CCN(C(c3cnc(=N)[nH]c3)=O)C2)ccn1 C(=O)(N=c1cc[nH]c(C)c1Cl)NCCS(CC)=O O=C1CCC(S(=O)(=O)NCC2COCCN2C(c2c(F)ccnc2Cl)=O)CC1 C1(CC=C)(NC(=O)CNC(C2CC23CC3)=O)CCCN(C(C2CCCO2)=O)C1 c1(C(=O)NC(C)C(=O)NCC2CCSC2)ccc(=N)[nH]n1 c1(COCC)nc(C)c(C(=O)NCC(C2(C(F)F)CCCO2)=O)s1.C1(C)(C)CN1 C1(C(=O)NC2CN(c3ncco3)C2)CCN(C(C2CC(=O)N2)=O)C12CCC2 N1(C(c2[nH]cc(S(=O)(=O)N(C)C)c2)=O)CCCCCCCCCC1 CC(C)(C)S(=O)(=O)c1ccc(NCCC2COCC2O)cn1 c1(C(N2CCN(C(C=Cc3nnn(C)n3)=O)CC2)=O)ncc(C(F)(F)F)cc1Cl c1(NCC2CN(C(C(c3ccccc3)OC)=O)CC2C)ncccc1[N+](=O)[O-] c1(C(=O)NC(CCOC)CNC(c2ccc(C)s2)=O)c(SC)cccc1F N1(C(C=Cc2cc(C)no2)=O)C(C)CN(C(c2nn(C)nc2C)=O)CC1C O=S(=O)(c1ccc(Br)cc1)N1CCN(CCNC2(CO)CC3(CC(F)C3)C2)CC1 N1(C(CSc2n(C)ccn2)=O)CC2CCC(NC(C3(CO)CCC3)=O)CC2C1 Cc1nc(NC(C2CCCN(C(=O)CC(C)(C)O)C2)=O)c(F)c(Cl)n1 C(=O)(C#CC(C)(C)CNC(=O)C(C)C(F)F)NCCCOC=C N1(C(C(C)Cc2ccco2)=O)CC2CC(O)C1C2NC(c1ccc(N)cn1)=O c1(CC)ccc(C(=O)N(C)CC2CN(C(C3CNC(=O)C3)=O)CCO2)cn1 CC1COCC(C(=O)NC2CC(CNC(c3ccncc3C(F)F)=O)C2)O1 N1(C(Cc2onc(C)n2)=O)CC2CN(C(=O)CCc3ccc(F)c(Br)c3)CC12 C1(COC)CCCN1C(=O)CCCC1(NC(=O)C(n2cc(C)cn2)C)CCC1 N1(C(C(CC)C2CCC(=O)N2)=O)CCN(C(C2CCCCN2C)=O)CC1C C(c1cc(F)cc(F)c1)=CC(=O)NCC1CC(OC)CN1C(C1CC(OC)C1)=O C1(C)(C(=O)NCCOCCNC(C2CC(C)(C)C2)=O)COCC1(F)F C1(C(=O)NCCC2CN(C(c3c(OC)c(Cl)sc3)=O)C2)CCCC1C1CC1 Cc1csc2ccc(C(=O)NC3CC3NC(=O)C(F)=C3CCC3)cc12 C(=O)(C#CC1CCCCO1)NC1C(SC)CN(C(c2ccnc(O)c2)=O)C1 C=CCC(CC=C)C(=O)N1CCC(CNC(=O)C(C2CCCCCC2)O)C(C)C1 CC(CCCCN)NC(=O)Nc1cccc(C(c2ccc(O)cc2)=O)c1 C1(C(=O)NCC(CC)N(C(=O)CN2CSCC2=O)C)CCC(=O)N(CC)C1 N1(C(c2cnn(CC)c2C)=O)CC2CC(C1)C2NC(C1CN(S(N)(=O)=O)C1)=O N1(C(c2nc(CC)sc2)=O)CCC(C(C)NC(=O)COCC2CCOC2)CC1 CCCCC(C(=O)NCCCCCN(C)C(C12COC(CCO1)C2)=O)NC(N)=O C1(C(=O)NCCCCN(C)C(C2CC3CC3C2)=O)CCC2CC2CC1 C1(CN(C(c2cnc(C)o2)=O)C)COCCN1C(=O)CC1CNC(=O)C1 N1(C(C2(CN3CCCCC3)CC2)=O)CCC(F)(CNC(C2(c3cccs3)CC2)=O)C1 CC1CCC(C(=O)N2CCn3cc(nn3)C2)CC1.c1(O)ccccc1F.C1CC1 CC1(C(=O)NC2CC(C(N3CC4(CSC4)C3)=O)CC2O)CC2CC2C1 C(=O)(C1CCCn2ccnc21)NC(CNC(c1n[nH]c(CC)c1Cl)=O)(C)CC c1(C(=O)OC)cccc(NC(C2(C)CCCN2C(c2ccncc2Cl)=O)=O)n1 N1(C(Cc2cc(C)sc2C)=O)CCC(C2CCN(C(c3c(C)noc3N)=O)CC2)C1 c1(NC(C2(C)CCN2Cc2c(F)cccc2F)=O)nc(C(F)(F)F)cc(Cl)n1 CC(C)C(F)C(=O)NCC1(C(=O)NCC2CCCCC2)CC=CC1 CCCC1C(=O)N1.C1(C(N2CC(CO)C2)=O)CCCN1 Cc1c(C(=O)N(CC(O)CNC(C2CCCCS2)=O)C)c(C(F)F)nn1C C1(CNC(c2c(C)n[nH]c2)=O)CC12CCN(C(c1csc(C)c1C)=O)CC2 CCN(CC(=O)NC(C)COC(C)C)N1CCCC(C(=O)NC)C1 c1(C(N2CCC(CN(C(=O)C(F)CC3CCC3)C)C2)=O)cnc2c(c1)ncn2C CC1CC(NC(C2(c3cncc(F)c3)CC2)=O)CN(C(=O)CN(C2CCC2)C)C1 N1(C(c2cc(C)on2)=O)CCCC(C(C)(C)C(=O)NCC2COCCO2)C1 CC1CC2(CC(C(N3C(CNC(=O)Cc4cc(C5CC5)on4)CC4CC34)=O)C2)C1 c1(C(=O)NC2C(NC(=O)Cc3ccc(Cl)cc3Cl)CCC2)ccc([N+](=O)[O-])cc1 C1(NC(C(c2ccn(C)c2)C)=O)CCCC2CN(C(C3CCC3)=O)CC12 c1(C(N2CCC(CCNC(C=CC(CC)C)=O)CC2)=O)cc(Cl)c(Cl)cc1OC c1(NCC)ccc(Cl)c(C)c1Cl.c12ccc(cc1)C(=O)N1CCC1C(=O)N2C c1(C(N2CC(C=C)C(NC(=O)CCCCOC)C2)=O)cccc(S(=O)(=O)NC)c1 C1(C(=O)NC2CC(N(C(CC(C)c3cccnc3)=O)C)C2)CC(=O)NC(=O)N1 CCC(CC(=O)NCC1(CNC(C2(CCOC)CC2)=O)CC12CCC2)OC Cc1cc(NC2CCC2c2ccc(F)cc2)ccn1 C(=O)(C1c2c[nH]nc2CCC1C)N1CCC(CC=C)(NC(=O)C=CCCC)CC1 Cc1ccn(C(C)CC(=O)N2CCCC2CCCNC(c2sccc2F)=O)n1 c1(CC(=O)NC23CC(C2)N(C(=O)CCCn2cccn2)C3)ccc(F)c(Cl)c1F CCCCC(O)C(C)C(=O)NCCC(O)CNC(=O)C=C1CCN(C)CC1 c1(COC2CN(C(C34CC(C(=O)OC)(C3)C4)=O)CC(C)C2)ccc2c(n1)CCC2 C#CCC(C)(C)C(=O)NC(c1ccc(F)cc1)CNC(=O)Cc1c[nH]nc1O c1(OC)cccc(C(N2CCC(NC(c3ccnn3C3CC3)=O)C2C2CC2)=O)c1 N1(C(C(COC)OC)=O)C(C(=O)Nc2cnc(OC)nc2)CCC12CC2 N1(C(C(C2CCN(C(c3ncc(C)c(C)c3)=O)C2)(C)C)=O)CCC(C)CC(C)C1 c1(NC(c2c(C)oc(C3CC3)n2)=O)ccc2c(c1)CCC(N)C2 C1(NC(c2cn(C3CC3)cn2)=O)CCN(C(c2ccccn2)=O)CC1CO C(=O)(C(O)C(F)F)N1CCC(CN(C(=O)Cc2cccc(Br)c2)C)C1 C1(C(N2CCC(C(=O)NC(CNC(=O)OC)C)C2)=O)C2CCC(C2)C1C C1(C(=O)OC)CCN(C(=O)C(c2n[nH]cc2Br)N(c2ccc(Cl)cc2)C)CC1C C1(NC(=O)COC2CC=CC2)CCCC1CNC(=O)C(O)c1cnc[nH]1 C(=O)(CCC(C)(C)F)NCc1ccc(-n2cc(-c3cc(C(C)C)no3)nn2)nc1 C(=O)(C(C)CS(C)(=O)=O)NCC(C)NC(c1cc(C(N)=O)ccn1)=O O=C(N=c1[nH]nc(Cl)cc1Br)c1ccc(Cl)nc1NCc1cccc2ccnn12 C1(F)(C(=O)NC(CC)CNC(=O)C=CC2CCCO2)CCC(=O)CC1 N1(Cc2c(C)cc(C#N)cc2C)CCS(=O)(=O)C2CCCC12 C(c1ccc(Cl)s1)=CC(=O)N(CC)CC1CCCN1C(=O)Cc1nc[nH]n1 n1(CC)ncc(=NC(=O)C2(C)CCC(c3nc(C)no3)O2)[nH]1 C1(C(=O)OCC)(SCC(=O)NCC2C(NC(C3CCCC3)=O)C2C)CCCCO1 C=CCC(C(=O)NCc1ncn(C2CC2)n1)NC(c1c[nH]nc1COC)=O c1(C(=O)NCCC2CC2)csc(CNC(=O)C(F)C2CCOC2)c1 C1(CC)CN(C(C2CC2c2sccc2C)=O)CCC1NC(C1(SC)CC1)=O n1(CC(=O)NC2COC3(C2)CN(C(c2cscn2)=O)C3)cc([N+](=O)[O-])ccc1=O N1(C(c2n[nH]c(C(C)C)c2Br)=O)CCCC(NC(c2ccnn2C)=O)C1C C(=O)(C(C(C)C)NC(c1ccco1)=O)N1CCC(CNC(CCNC(C)=O)=O)C1 Cc1nnc2n1CC(C(=O)NCCCC(C)NC(=O)C=Cc1ccco1)CC2 c1(C(N2CC3C(CNC(c4cccnc4S)=O)C3C2)=O)cc(F)c2[nH]nnc2c1 C1(C(=O)NCCn2ccc(C(=O)NC(CO)C3CC3)c2)C2CC3C(C2)C13.CC C(=O)(C(C)CC=Cc1ccccc1)NC(c1ccccc1)CNC(CCC=C)=O C=CC(C)(CCOC)C(=O)N1CCN(C(c2ccc(C3CC3)nc2)=O)CC(C)C1 C1(C(=O)NCC(N(C(CC)=O)C)C2CC2)CSCCN1C(=O)OC(C)(C)C C12(CC(=O)NCC3(C(=O)OC)CCC3)CCC1CN(C(=O)C(C)c1cc[nH]n1)C2 C(=O)(CC(O)CC(C)(C)C)N(C(CC)CC(=O)NCc1oc(C)nc1C)C CCCCCC(F)C(=O)NC1(CC(=O)NC2CCCCC2C)CC1 C(=O)(C1c2ccccc2C2CC1C2)N1CC(NC(=O)COC(F)(F)C(F)(F)F)C1 C(=O)(C(C(=O)N1CCC(NC(=O)C=CSC)C1)C(C)(C)C)OCC [N-]=[N+]=NCCCC(=O)N1CCCC1C1CCN(C(C2(n3cccn3)CC2)=O)CC1 C(=O)(CC(C)(C)C(F)F)NC1C(CC(=O)NCc2cc(C)on2)CCCC1 C1(C)(NC(C)=O)CCN(C(=O)CC(C2CC2)NC(=O)Cn2cncn2)C1 C1(Cc2ncc(C(N(C)NC(CC(C)OC(C)(C)C)=O)=O)o2)CC2(CC2)CO1 c1(OC)ccc(C(C)C(N2CC3CC2C3CNC(=O)C(F)(F)C2CC2)=O)cc1 C1(C(=O)OC)CC2CC(C1)CN(C(C1CC1c1ccc(O)c(Br)c1)=O)C2 C1(CC)CC(N=c2nc(N3CCC4(COC(C)C4)C3)c3ccccc3[nH]2)C1 C(CC1=CCCCC1)NC(C(c1ccoc1)NC(Cc1c(C)nsc1)=O)=O c1(CC(=O)N(C)CC2CN(C(Cc3c(C)scc3)=O)C2)ccc(C(N)=O)cc1 C12(C(=O)NCC(CNC(C(CC)NC(N)=O)=O)O)CCCCC(F)(C1)C2 Cc1c(CC(=O)NCC2(C)CN(CC3CCC(C(F)(F)F)CC3)C2)cnn1C n1(CCSC)nnnc1C(c1ccn(C(C)C)n1)NCc1cc(Br)co1 CCCCC(C(=O)NC1CC1NC(c1cnc(Br)c(O)c1)=O)N(C)C C=CC1(NC(C(=O)O)C2CN(C(=O)OC(C)(C)C)C2)CCCCC1 CC1=NNC(=O)C1CC(N1CCCC1C(C)(C)C(=O)N(C)CC1(CO)CC1)=O Cn1nnc2cccc(C(=O)NCCC3CN(C(c4cc(Br)no4)=O)C3)c12 CC1c2ccc(Cl)cc2CCN1C(=O)CCc1ccsc1 Cc1cnc(N2CCN(C3CCN(C(C4(C)CCCS4(=O)=O)=O)C3)CC2)nc1O N1(C(CCCOC(C)=O)=O)CCCC(C(C)NC(=O)CCc2cc(C)n(C)n2)C1 Cc1cccnc1C=CC(=O)NC1(CC(=O)NC(C)CN(C)C)CC1 c1(C(N(C2CCN(C(C(C=C)C)=O)C2)CC)=O)cc(=O)c(OC)c[nH]1 N1(C(C(N2CC(C)C2)C)=O)CCC(NC(C2CC(OC(F)F)C2)=O)C1 N1(C(C23N(C(C4CCCC(C)CC4)=O)CC(C2)C3)=O)CC2(CCCN2C)C1 C1(N(C(C2C(C)C2)=O)C)CC2CCC(C1)N2C(=O)C(c1cccc(F)c1)O N1(C(C(C)NS(C)(=O)=O)=O)CCC(C(C)(C)NC(c2ccncc2)=O)C1 C1(NC(CC(N)C2CCCC2)=O)CCN(CC)CC1O.C(C(F)(F)C(F)F)OC=O C12(C(N3C4CN(C(CCC(C)SC)=O)C(CC4)C3)=O)CCCC(=O)N1CCC2 N1(C(C(CC2CN(C(C(CC)C#N)=O)C2)F)=O)CC2CCOC(=O)C2C1 C(=O)(C(CC)C(C)(C)CC)NCC12CC(CNC(CC=CC)=O)(OC1)C2 C(=O)(CC1=CCCCC1)NC1(CC=C)CN(C(=O)C(c2ccncc2C)C)C1 C=CCC(CC(C)C)C(=O)N1CC2CC2(CNC(C2CCN2C2CCCC2)=O)C1 c1(C(C(=O)NC2CCC2)NC(C=CC=CCC)=O)ccccc1 CCCCC(O)C(C)C(=O)NC1CC(CC(N2CCCC2CSC)=O)C1 N1(C(CCOCC)=O)CCCC(CNC(=O)C(C)(C)CC2CC2)CC1 C(=O)(C#CC1CCCCC1)N1C(C)CCC(NC(=O)C=CC2CCOC2)C1 C1(C(=O)NCC(C)NC(COC(C)=O)=O)CCCN1C(c1cccs1)=O C1(NC(c2c(C)cncc2)=O)(CNC(=O)CCc2ccncn2)CCCCC1C C1(C(N(CC(C)C(=O)NCCN2CCC(CO)C2)C)=O)CCOC(=O)CC1 C1(C(=O)NCC(CC)NC(C2(SC)CC(F)(F)C2)=O)CCN(C)C1=O C(=O)(CCC#Cc1ccccc1)NCCN1CCN(C(C=CC(C)(C)C)=O)CC1 c1(C(N(C)CC2CCN(C(=O)CC(F)F)CC2)=O)ccc2nc(S)[nH]c2c1 c1(CNC(C2N(Cc3ccc(C(N)=O)nc3)CCC2)=O)ccc2cccnc2c1 N1(C(C(C)OC)=O)CCCC(C)(C)C1CNC(c1cccn2cncc12)=O C1(C(C)C)CN(C(c2ncnn2C)C(=O)Nc2ccc(Br)cc2)CCO1 Cc1ccc(SCC(=O)NCC2COCC2NC(=O)COC2CCOCC2)cc1 C1(F)(C(=O)NC(C#C)(C)C2CC2)CCCN(C(=O)Cn2nccn2)C1 c1(C(=O)NCCC2CCN(C(COCCOCC)=O)C2)ccc2ccsc2c1 C(=O)(C#CC1CCCCC1)NC(C1CCCCN1C(=O)CCc1ccccn1)C CC1CC(NC(=O)CC2(C3CC3)CC2)CCN1C(=O)Cn1cccc1 CC1C(NC(c2ncc[nH]2)=O)CC2CCC1N2C(c1cnn(C(C)(C)C)c1N)=O C(CNC(c1ncccc1F)=O)(C(C)C(C)C)NC(c1c(C)ncnc1)=O C1(C(=O)NC2CC(CC(=O)N(C(CC(CC)C)C)C)C2(C)C)CC2(CC(=O)C2)C1 C1(CC=C)(NC(=O)C(N2CCC(C)C2)=O)CN(C(C2CC2C)=O)C1 N1(C(C(CC)C)=O)CC(C2CCN(C(=O)CC3C(C(=O)OC)C3(C)C)CC2)C1 C1(C(N2CC(O)(C(C(=O)NCc3nc(COC)on3)F)C2)=O)CC12CCCCC2 S(=O)(=O)(c1cccs1)N1CC(C(N2C(C(=O)OCC)CCC2)=O)C1 c1(CN(c2cccnn2)C(C2CCCN(C(C)=O)C2)=O)c(Cl)oc2ccccc12 C1(C(=O)NCCC(C)NC(C2CC(=C)C2)=O)CCCN(C(=O)OC)C1 CCC(C)(C)C(O)C(=O)NCCC1CCN(C(c2occ3c2CCC3)=O)CC1 N1(C(C(CCSC)O)=O)CC2CC(NC(=O)CCC3CC(F)(F)C3)CC1C2 C1(C)(CCNC(CCC=C(C)C)=O)CCN(C(=O)C=Cc2ccc[nH]2)C1 C12(C(N(CC(O)CO)CC)=O)CC(CO1)N(C(=O)C=CC1CCCC1)C2 C1(C(=O)NCCCCCC=C)N(C(=O)C(F)CCC)CCCC1(C)C O=C(C#CC1CCCCC1)NCCOC1CCN(C(c2c(O)cccc2F)=O)C1 C1(C(=O)NC(C)CCCCNC(c2cc(C#N)c[nH]2)=O)CC12CC(F)(F)C2 C(=O)(CC1=CCCCC1)NC1C(CC)N(C(=O)C(C)CC2CCC2)CC1 N1(C(CC2N(C(C)C)CCC2)=O)CCCCC(NC(C2C3CCC2CC3)=O)C1 N1(C(C(C)=CC2CC2)=O)CCCN(C(C2CCC(CN(C)C)CC2)=O)CC1 Cc1scc(C(=O)NCC(C)N(C(=O)C=CC(C)C)C)c1C c1(C(C(N2CCCC(c3cn(CCCCOC)nn3)C2)=O)O)c(C)cccc1C CCC(F)(F)C(C)(C)C(=O)NCC1(C)CCCN(C(=O)CCn2ccnc2C)C1 c1(C(=O)NC(CNC(C(C=C)(C)CC)=O)(C)C2CCC2)cc(F)c(F)c(C#N)c1 c1(OC)ccc(C(=O)NC(C)(CNC(=O)COCC(C)C)C2CC2)c(C)c1 C(=O)(C(CO)C(C)(C)C)N1CC2C(NC(c3nc(C(C)C)sc3)=O)C2C1 C1(CNC(C2N(CCC)CCC2)=O)CN(C(=O)CCCSC)CC(C)(C)C1 N1(C(C2CC(O)(CC#C)C2)=O)CCC(O)CC1C(=O)NC(C=C)CO c1(C(=O)NCCOCCNC(CCc2cc(C)[nH]n2)=O)cc2c(nn1)OCCS2 c1(CNCC2N(C(c3scc(N)n3)=O)CCOC2)c[nH]c2cc(Cl)ccc12 C(C(CC(C)C)C(=O)NC(C)C(CO)NC(=O)CCN(CC(F)(F)F)C)OC Cc1c[nH]nc1Cn1cc(CNC(C2(CF)CC2)=O)nn1 C1(C(=O)NC2(CC#C)CC2)CN(C(C2CC(OC(C)=O)C2)=O)CC1F N1(C(c2c(SC)csc2)=O)CCC(NC(=O)CC(C)c2ccccc2)C12CC2 C1(C(=O)NC2CCC(C)(C)CC2)CN(C(C2CCC(=O)C2)=O)CC12CCC2 CC(CN(C)C)CCC(=O)N1CC(NC(=O)C=Cc2cn(C)nn2)C1 C1(C(=O)NCc2c(C)cco2)CCN(C(=O)CCC=CC(C)C)CC1(C)C C1(ONC(=O)Nc2cc(F)ccc2Br)CC12CCc1ccccc12.C12CC13CC23 c1(NCC(CNC(c2c(OC)cc(F)cc2)=O)C)ncnc2scc(Br)c12 Cc1cc(CNC(c2ncc(-c3ccc4nc[nH]c4c3)cn2)=O)cc(C)c1F C(=O)(N=c1nc2ccccn2[nH]1)N1CC(C)N(Cc2ccccc2)CC1 O=C1OC2CC1N(C(=O)NC1CCN(C3CCCC3)C1)C2 c1(C(N(C2CCN(C(=O)C(C3CC3)OC)CC2)CC#C)=O)cn(C)c(=O)c(C)n1 c1(NC(N2C(C(N3CCC(C)CC3)=O)CCC2)=O)cncc([N+](=O)[O-])c1 c1(C(C(=O)N(C)CC2CNCC2(F)F)O)cccc2c1OC(F)(F)O2 C1(NC(CN(CC)CC)=O)CN(C(=O)C=Cc2csc(Br)c2)CC1(C)C c1(C(N(C2CCN(CC3CCSC3)CC2)CC#C)=O)ccc2c[nH]nc2c1 c1(C(=O)NCCOCCN(C)C(C2CCO2)=O)cccc(C(=O)C2CC2)c1 N1(C(CC(C)C)=O)CCN(C(c2cc3nc[nH]c3cc2F)=O)C(C)CC1C CC1(C)COC(=O)C1n1cc(C2(F)CN(C(=O)Cc3cc(C4CC4)on3)C2)nn1 C1(C(N2CCC(N(C(C=CCC)=O)CC)C2)=O)CCCCCC1(F)F C1(O)(CC)CCCN(C(=O)C(Cc2cnc[nH]2)NC(c2cc(C)c[nH]2)=O)C1 N1(C(CC(C(=O)OC)C)=O)CC(C2CN(C(c3cc(C)cnc3C)=O)C2)C1 O=C(C1=CCOCC1)NC(c1cc(F)cc(Cl)c1)CNC(c1ccc(CO)o1)=O CCC(CC)C(F)C(=O)N1CCN(C(=O)C(CO)N(C)C)C(CCO)C1 C1(C(N2C(CNCC#C)CCC2)=O)CCN(C(c2coc(SCCC)c2)=O)CC1 C1(n2cc(CN3CC(C)C(NC(=O)CCCC(N)=O)C3)nn2)CNC(=O)C(C)(C)C1 C(=O)(C1=CCN(C(=O)CCc2cnn(C)c2)CC1)NC1C(CC)CCCC1 c1(C(C(=O)NCC(C2CC2)NC(C2(OC)CCCC2)=O)(F)F)ccc(F)cc1F n1(CC)cc(CC(=O)NC(C)CC2CN(C(=O)C(C)C3CCCO3)C2)cn1 c1(C(=O)NCCN(C(c2ncc(C)cc2C)=O)C2CC2)cnc2scnc2c1 N1(C(C2(CC=C)COC2)=O)CCOC(CN(C(=O)C(C)(C)C)C)C1 CN1CCCC1CNC(c1cc(CNC(c2ccncn2)=O)on1)=O C1(CCC)CN(C(=O)OC(C)(C)C)CCN1CCN1CCC1 CC1CCN(C(=O)C=CC(C)(C)NC(C2CCOC2)=O)CCS1 C(=O)(C1=NOC2(CCC2)C1)NC1CCC(NC(c2ccc(SCC)nc2)=O)CC1 c1(SCCCCCCNC2N(C)CCCC2)cccc(Br)c1F C1(C(N(C)Cc2c(C)c(Cl)ccc2)=O)CCS(=O)(=O)C(C)C1 N1(C(=O)CCCF)CCCCC1.c1(-c2c[nH]nn2)cncc(Br)c1 C1(N(C(=O)C=CCN2CCOCC2)C)CCC(NC(C2CCCOC2)=O)CC1 C1(C(=O)NC2(C)CCCN(C(c3ccc(F)o3)=O)C2)CCOCC12CCC2 C12CC(C13CCC3)NC2=O.N1(CC)CCC(C(=O)NCc2sccc2CSC)CC1 N1(C(C2C(C)(CC)C2)=O)CC2CC1C2NC(c1cnc(C)cn1)=O C1(NC(C(C)OC)=O)CCc2onc(C(=O)Nc3ccccc3[N+](=O)[O-])c2C1 Cc1ccc(C=CC(N2C(C(=O)N(CCO)C3CC3)CCC2C2CC2)=O)cc1 c1(NC(C2N(C(c3c(C)noc3C)=O)CCSC2)=O)cc(Br)cnc1C(N)=O C(=O)(C1CCCn2nccc21)NC(CN(C(C(CCCC)C)=O)C)C c1(C(=O)NCCC(C)N(C(=O)CS(N)(=O)=O)C)sc2cc(F)ccc2c1Cl CC1(C)CC(CNC(=O)CCNC(N)=O)N(C(=O)Cn2cc(F)ccc2=O)C1 C1(CNC(CC2CC(=C)C2)=O)CC(F)(CNC(c2ccsc2OCC)=O)C1 C(=O)(CCCCCC#N)NC1(C(=O)NCC(CC)(C)C)CC(CO)C1 C1(C(=O)OC)N(C(=O)C(C)CCc2ccc(OC)cc2)CCC1(C)C CCC(C)CC(=O)NCC(c1ccc(N(C)C)cc1)NC(=O)Cc1cncs1 C1(C(=O)NCCCCNC(c2cc(C)c(=N)[nH]c2)=O)CCn2cnnc2C1 C1(C)(C(=O)NC(c2cccnc2)C(=O)N(CC(C(=O)OC)C)C)CNC(=O)C1 Cn1ccc(=NC(=O)CCC2CCCN2C(c2cc(Cl)nc(Cl)c2F)=O)[nH]1 N1(C(c2nc(OC)oc2)=O)CCCC1C1CCCN1C(c1ccc(C)c(C)c1)=O Cc1csc(C(C)C(=O)NC2CC(C)(NC(c3cnns3)=O)C2)n1 CCC(CN(C)C)CC(=O)N(C)CCNC(c1ccc(Br)c(O)n1)=O c1(C(=O)NCC(CNC(C(C)N(C(C)=O)C)=O)CO)cnn2cc(C#N)cnc12 N(C)(S(=O)(=O)N(C)C)CC(N1CCN(CCNC(CC(CC)O)=O)CC1)=O c1(C(=O)NC2(CF)CN(C(c3c(C)con3)=O)C2)ccn(CCO)c1C CCC(COC)(CC)C(=O)NC1CCN(C(=O)Cn2nc(O)ccc2=O)CC1C NS(=O)(=O)N1CCCC(C(=O)NC2(CNC(C3(O)CCCCC3)=O)CCOC2)C1 c1(CNC(CC(OC)OC)(C)c2nnnn2C2CC2)ccc(C)c(C)c1 C1(CNC(=O)NC(c2cc(C3CC3)on2)C)C2C=CC(C2)N1C(=O)OC(C)(C)C O=S(=O)(c1cccc(=NCC(F)C2CCCC2)[nH]1)N1CCC(c2ccncc2)C1 c1(C(N2CC(NC(CN(C(C(C)C)=O)C)=O)C(O)C2)=O)cc(Cl)cnc1O c1(C(N(C)CC2CCCN2C(C2CC2C(F)F)=O)=O)cccc2sccc12 C1(CC(=O)NCCC(C)NC(C2CN(C(N)=O)C2)=O)CCOC1(C)C CCCCCC(C)CC(=O)N1CC(OCC(=O)NC2CC(C)(CC)C2)C1 CC1=NOC(C)(C(=O)NCC2CN(C(c3csc(C)c3C)=O)CCO2)C1 Cc1noc2ncnc(NC3CCN(C(=O)CCC(C)(C)C)C3)c12 c1(C(N2CCN(C(CNC(=O)OCC)=O)C3C2C3)=O)cc(F)cc2c1NCCC2 N1(C(Cn2nc(C)c(Cl)c2C)=O)CCN(C(c2cccc(=O)n2O)=O)CCC1C Cc1ccc(C(=O)NCC(O)CNC(c2ccc(Cn3ccnn3)o2)=O)o1 C1(NC(c2cc(C(=O)OC)no2)c2nnnn2-c2ccccc2)CCN(O)C1=O.C1CC1 c1(OC)cncc(C(=O)NCC2(NC(=O)CCCOC(C)C)CCCCC2)c1C Cc1nc(=N)[nH]cc1C(=O)NCC1CCC1NC(c1ccnn(C)c1=O)=O c1(C(=O)NC(CC)(C)CNC(C2CCC(C)C(C)C2)=O)ccc2nccnc2n1 Cc1cnccc1C(=O)NCCN1CCN(C(C2(C)CC2C)=O)CC1 N1(C(C2C(CC)OCC2)=O)CCCCC(NC(c2ccc(O)c(Cl)n2)=O)C1 C1(NC(c2c(CC(=O)OC)cccc2)=O)CCC(C)N(C(c2csnc2C)=O)C1 C(C)(c1ccc(CC)cc1)=CC(N1CC(CNC(COCCC=C)=O)C(C)C1)=O c1(N2CCC(CC(=O)NCCSc3ccccc3Cl)C2)ccc(N(C)C)cn1 c1(C(CC)(CC)NC(=O)CC23CC(C2)C3)ccc(Br)cc1 c1(C(N2CCC(OCc3ccccc3)C2)C(=O)NCC)cccc(C(=O)NC)c1 C1(CC(=O)N(CC(C)O)C)(NC(=O)CC(N)c2ccccc2)CCOC1 C1(C2CCN(C(C3CCCNS3(=O)=O)=O)C2)(NC(c2c(CC)cco2)=O)CC1 C1(OC)CC2CCC1CC2C(=O)NCC1(F)CC(CNC(C2SCCC2C)=O)C1 N1(C(C2(CSC)CC2)=O)CCC(CCC(=O)Nc2ccccc2F)CC1 c1(-c2c(Cl)ncc(C)c2)ccc2c(C(N3CCC(C4COC4)CC3)=O)n[nH]c2c1 C=CCCN=C(NCC1CCN(C)C(=O)C1)N1CCCCC1 c1(C(=O)NC2CC(CCNC(C3C(OC)CCCC3)=O)C2)cc(Cl)cc(C)c1N N1(C(c2cc(C)[nH]c2)=O)CC(NC(=O)CC2CCOC2)C2CCCCC12 N#CC1(CN2CCCC(N)(C#N)C2)CC2(CCC2)C1 Nc1sc2c(c1C(=O)NCC1CCCC1NC(=O)C(O)CC1CC1)CCC2 C1(NC(=O)COC(F)F)CCSC12CN(C(c1cc(C3CC(F)(F)C3)[nH]n1)=O)C2 c1(C(=O)OC)cc(C(=O)NC2CN(C(C3CC4(CSC4)C3)=O)CC2C)ccc1F c1(C(C(=O)Nc2n[nH]c(C)c2-c2cccc(Cl)c2)O)ccc(C#N)cc1 CC(=O)CCN=C(NCC1COC(C)(C)O1)NC(C)CC(C)(C)C N1(C(CC)=O)C2CCC1CC(NC(c1cc(OC)nc(Cl)c1)=O)C2 N1(C(Cc2ccc(OC)nc2)=O)CCC(NC(c2c(Cl)sc(C)c2C)=O)C(O)C1 N1(c2nc(COC)nc(O)c2)CC2(CN(C(=O)Cc3ccn(C)n3)CC2CO)C1 c1(C(=O)NCCNC(c2cccc(NC(=O)OC)c2)=O)ccc(F)c(N)c1 C1(C)(C(N2CC(CCNC(C3CCC3c3nc[nH]n3)=O)(OC)C2)=O)CCNC1=O c1(C(=O)NC(C(C)NC(CSCC(C)C)=O)CO)cc2ccccc2s1 Cc1ccc(C(=O)NC2CCC2NC(=O)COC2CC2)cc1Br N1(C(C(C)(C)OC(C)=O)=O)Cc2nccn2CC(NC(=O)CC(C)N(C)C)C1 C(CC(=O)NC1CCOCC1O)(C(F)F)NC(c1c(C)oc(CO)c1)=O Cc1nc([N+](=O)[O-])cn1CC(=O)N(CC(C)CNC(=O)CN1CCC(C)(O)C1)C c1(OCC(=O)NC(CC(C)NC(C2CC(=C)C2)=O)C)ccc(C)cc1 C1(CNC(c2cc3n(n2)CCC3)=O)CCC12CCN(C(C1CCOC1)=O)CC2 c1(C(N2C(CCNC(COC(C)C)=O)CCCC2)=O)cccc2c1CCOC2 c1(OC)cc(O)ncc1C(=O)NC1(C)CN(C(c2cccnc2OCCO)=O)C1 C1(OC)CC(NC(=O)C(C)NC(N)=O)CN(C(=O)Cc2ncn(C)c2C)C1 c1(C(=O)NCCCCCNC(Cc2ccn(CC)n2)=O)ccc2c(n1)CCCC2 S(=O)(=O)(c1cc(Cl)c(Br)cc1F)N1CCC2(CC(NC(c3ncsc3Br)=O)C2)C1 N1(C(c2cnc(C)n2C)=O)CCN(C(c2cccnc2O)=O)C(C2CC2)C1 C(CCCC(F)(F)C(F)(F)F)NCc1ccc(C(=O)OCC)s1 C1(Cn2cc(C=CC)nn2)CCN(C(C2(C#N)CCCC2)=O)CC1(F)F C(=O)(C1=CC(C)(CC)C1)N(CCCNC(C(C=C)(C)C)=O)CC1CCCC1 C1(NC(=O)CC2CNC(=O)O2)CCC(NC(C2(CF)CC(F)(F)C2)=O)CC1 CCC(C(=O)NC(C)C(F)(F)F)NC(=O)C=C1CCCC1 N1(Cc2nnc(C(C)(C)C)s2)C2CCCC1COC2 C1(CNC(c2c(C)cc(C)c(C)c2)=O)CCC2(CCC2)CN1C(c1cnco1)=O N1(C(c2cnn(C(C)C)c2F)=O)CCC2CCC12CNC(=O)CCC(N)=O Cc1nn2ncccc2c1C(=O)NCC(C)(C(C)C)NC(=O)C=Cc1cncs1 C(=O)(C1=CS(=O)(=O)CCC1)N1CCCC(N(C(COC(CC)C)=O)CC)C1 CCC(C(=O)N(CCNC(c1c[nH]cc1Br)=O)C1CC1)Oc1ccccc1 N1(C(CCCCCOCC)=O)CC2(C)CN(C(=O)CN3CCC3)CC2(C)C1 C1(C(=O)NCC2(F)CN(C(C(C)(C)C)=O)C2)COc2ccccc2C1 C1(C2CCC(NC3CCC(C)(C)C3)CC2)(C(=O)OC)CC1 C12(C(N3CCCC(O)(CCNC(C4CCCC4)=O)C3)=O)CC1Cc1c[nH]nc12 N1(C(=O)C(C)(C)OC(C)=O)CC2CC(NC(c3c(COC)noc3)=O)C2C1 C1(C)(C(=O)NCc2c(C(=O)NC(C)(C(C)OC)C3CC3)nco2)CCOCC1 c1(C(=O)NCC(C2(O)CN(C(C(=O)NCCOC)=O)C2)(C)C)c(C)cccc1Cl c1(C(=O)NC(C)CCC(N2CCCC(C)C2CO)=O)ccc2ccncc2n1 c1(OC)cc(CNC(C2(C)CN(C(=O)Cn3ccnn3)C2)=O)cc(F)c1 CN1CCOCC1C(N1CC(CNC(C2(N3CCCCC3=O)CC2)=O)C1)=O C(C1CCN(C(=O)C=Cc2ccn(C)c2)CC1)=CC(=O)N(CCOC)CC N1(C(C2(C)CC2)=O)CCN(C(C2CCC3CC3CC2)=O)CC1CC(F)F C12(C(N3CCC(C)(F)C3)=O)CCC(CC1)N(C(c1ccsc1Cl)=O)C2 C1(CNC(C2CC(C#C)(O)C2)=O)C(C2CC2)CCN1C(c1ccc(CC)cc1)=O c1(CCC)nnc(S)n1CC(=O)NC(C)CCNC(c1ccn(C)n1)=O c1(NCC(N(C(C2CCN(C)C2=O)=O)C)C2CC2)ncnn2cccc12 C1(O)(CC(N2C(CNC(C3(C(=O)OCC)CCCC3)=O)CC2)=O)CCCOC1 c1(OCC(=O)OC(C)C(=O)NC2CCC(O)CC2)cc(Cl)cc(Cl)c1 C1(N(C(CCCC)=O)C(=O)Cc2nn(C)cc2Br)CC(F)CN(CC)C1 N1(C(CC2(C)N(C(c3scc(C)c3)=O)CC2)=O)CCn2c(C)nnc2C1 Cc1ncnc(C)c1NC(=O)C(CC1CCC1)OC(=O)CC(C)(C)CN(C)C N1(C(C2C(OC)CCCC2)=O)CCC(C)N(C(c2csnc2C)=O)CC1 c1(C(=O)NCCC2COCCN2C(c2cccnc2O)=O)cc2cn[nH]c2cn1 N=c1[nH]cncc1C(=O)NC1CC(CNC(=O)CC2CSCCS2)C1 C=CC1CN(C(=O)C(CC)CCC)CC1NC(c1ccc(CS(C)(=O)=O)cc1)=O C=CCCCCCCCC(=O)N1CCN(C(=O)C=Cc2cocn2)C(C)C1C C1(CNC(=O)COCCN(C)C)CC(O)CN1C(c1cnn(CC(F)(F)F)c1)=O CN1CCN(C(=O)C(CCOCCO)NC(c2n[nH]c(O)n2)=O)CC(O)C1 N1(C(C2=CC(C)(CC)C2)=O)CCC2(CCOCC2)C(NC(c2cc(OC)n[nH]2)=O)C1 N1(C(C)C)C(=O)COCC1C(=O)N(C1CCCN(C(=O)COc2ccsn2)C1)C CC(CC(=O)NC1CC2(C1)CN(C(=O)Cc1cccc(Cl)c1F)C2)CC(F)(F)F c1(CC)nc(C)[nH]c1C(=O)NC1CC12CC(NC(=O)CC(C)c1cnn(C)c1)C2 N1(C(C2(C)CC(C#N)C2)=O)CC23CCCC2(C1)CN(C(=O)C=Cc1cscn1)C3 C(=O)(CP(C)(C)=O)N(C1CCC(NC(=O)CCCC2CCCCC2)CC1)CC C(=O)(C1Cc2ccc(Cl)cc21)N1C(CNC(C2CCCCC2)=O)CC1 CC(CC(=O)OC(C)(C)C)c1cccnc1.C1CCCNC(=O)C2C(C2)C(=O)N1 c1(CNCC2(C(=O)NC(C)CF)CC2)c(Cl)ccc(Br)c1F Cc1ccc(CC(N2CCCC2CCCNC(C2CC(N(C)C)C2)=O)=O)cc1C N1(C(C2C(C#N)CC2)=O)CCCC(CCNC(c2c[nH]nc2C2CC2)=O)CC1 CCCC(C1CCC1)NC(C1CCC1CNC(=O)C=C(C)C(F)F)=O c1(CC(=O)NCC2CN(C(CCN(C)CCO)=O)C2)c(Cl)ccc(O)c1Cl N1(C(CN(C)CCO)=O)CC2CCC(C1)N2C(=O)Cc1ccccc1S(C)=O C1(CC)CCN(C(=O)Cn2cc(CO)nn2)C(C(=O)N2CCCCO2)C1 c1(C(=O)NCC(C)NC(c2ncc(C3CC3)cc2F)=O)c(Cl)ccc(O)c1N Cc1cc(Br)c(NC(C2CC3(C2)CN(Cc2cscc2Br)C3)=O)cc1C N1(C(C(C)(C)F)=O)CCC2(CCC(NC(c3ccn4nccc4c3)=O)C2)CC1 CC(C)CC(C(=O)N1CC(OCCNC(C2CCNC2=O)=O)C1)C(C)C C1(CN=C(NCc2nc(C)sc2)NC(c2ccccc2)C)CC(S(C)(=O)=O)C1 C12(C(N3C(CCC(C)(C)NC(C(C)C)=O)CCCC3)=O)CC(C)(C1)OC2C c1(C(=O)NC2(C)CN(C(C3CC(=O)C34CCCC4)=O)C2)ncn2ccccc12 c1(N2CCCCC(C)C2)nc(=NCC2(c3ccccn3)CCC2)[nH]c2c1SCC2 C(c1ccc(C(N)=O)o1)=CC(=O)NN(C(=O)C=C1CCCCC1)CCOC.C1(C)CC1 c1(C(N(CCCNC(COCCCCC)=O)C2CC2)=O)cnccc1OC(C)C c1(C(=O)NCC(C)(CO)NC(C2CC(Cl)(Cl)C2)=O)ccc2oc(O)nc2n1 N1(C(CS(CC(C)C)(=O)=O)=O)CC(NC(=O)CC2CC2)C2(CCS(=O)(=O)CC2)C1 Cc1cc(=NCCNC(C2CCCN(C(=O)C(O)C(C)C)C2)=O)nc(C(C)C)[nH]1 C(=O)(C1Cc2ccc(Cl)cc21)NC1C2(CCC(NC(=O)COC3CCC3)CC2)C1 N1(C(=O)NCC(c2c(C)cno2)=O)CC(C(F)(F)F)CC(SC(C)(C)C)C1 N1(C(C2(CCOC)CC2)=O)CC2CC2(CNC(C2(C)CC(F)(F)C2)=O)C1 C1(C(=O)NC(CC)CSC)N(C(C2CS(=O)C2)=O)CC12CCCC2 C1(C(=O)NC(COC)C(C)C)CNC(=O)CC12CCOC2 C(CC(=O)N1C(CO)CC1C)(C(C)(C)C)NC(C1=CCCC1C)=O c1(C(=O)NCC(CC)NC(=O)CCCC2CCC2)cccc2nc(C(C)C)[nH]c12 N1(c2ncc(C)c(O)n2)CC2(C1)C(NC(=O)C(C(C)C)N(C)C)CCS2(=O)=O Cc1nc(NC23CCC(CC2NC(c2nn(C)cc2Cl)=O)C3)ccc1C#N C(C(O)CC(=O)N1CCCC1CC1CC1)NC(C(n1ccc(C)n1)C)=O C1(C(=O)NCC(CSC)(C)O)(NC(C2CC3CC3C2)=O)CCCCC1 C1(C(N2CCC(C(C)NC(CCOC(C)C)=O)CC2)=O)CCN(C)C(C)C1 N1(C(c2c[nH]c(=NC)s2)=O)CCCN(C(c2cnc(C3CC3)nc2O)=O)C(C)C1 C(=O)(C1=CCCN(C(=O)C(C)CC2CC2)C1)NCC(CC)OC c1(C(N(C(C)CCNC(=O)Cc2cccs2)C)=O)cc(Cl)ccc1O c1(C(C)C(=O)N(c2nn[nH]n2)C(C2CNC2)=O)cccc(F)c1 C1(C(=O)OC)CC(n2cc(CSC)nn2)CN1C(=O)C(c1ccccc1)C C1(NC(C2(C(N(C)C)=O)CC2)=O)CC(C(=O)Nc2c[nH]ccc2=O)=CC1O c1(CC)c(C(=O)NCCCCCCNC(=O)CC23CCCC2C3)csc1C N1(C(C)C)CCC(NC(C2(NC(C3CC(C)CO3)=O)CCC2)=O)CC1 N#Cc1cccc(C(=O)NC2CCCC2NC(C2CCN(S(C)(=O)=O)C2)=O)c1F N1(C(C(C(C(C)C)O)(F)F)=O)CCC2(CCCN(C(=O)Cc3cccn3C)C2)C1 c1(C(C)C(=O)NCCNC(C2(Cl)CCCCC2)=O)cccc2ccccc12 c1(C(N2CC3(C(C(=O)OCC)C3)C2)=O)c(OC)cccc1F.C12CCCN1C2 Cc1cncc(C(N2CCCC2(C)C(=O)N(C2CN(C(C)C)C2)C)=O)n1 C1(OCCC)C(C)CCCN1N(Cc1cncs1)Cc1ccccc1F N1(C(c2cc(C)sc2)=O)CCC(N(C)C(C2CC2C#N)=O)CC1 C#CC1CCCC(CNC(=O)CC2C3CCC(C3)N2C(=O)CC(C)(C)C2CC2)C1 C(CCCCNC(=O)CC1(C)CC1(Cl)Cl)NC(C=CCOC)=O C=C(C)CC(C)C(=O)N1CCOCC1CNC(c1ccc(-c2ncon2)cc1)=O N1(c2[nH]c(N(C)Cc3cccc(F)c3F)nc(=NC)n2)CCOC2(CCSC2)C1 Cc1nc(C(N2CC=CC(NC(=O)CNC(=O)CCCCO)C2)=O)nn1C c1(NC(c2nccs2)C)nccc(=NC2CCC(F)(F)C2)[nH]1 CCC(C)(C)C(C)CC(=O)NCCOCCNC(c1ccc2snnc2c1)=O c1(CC)cc(C(N2CC(CNC(=O)C=C3CCC(C)CC3)(OC)C2)=O)ccc1F C#CCCC(O)C(=O)N1CCCC(C)(CNC(c2conc2COC)=O)C1 c1(NC(C)=O)ccc(Br)cc1C(N1CC(NC(c2ccnnc2C)=O)C1)=O CCCC(C)C(=O)NCCC1CC(OC)CN1C(c1cn(CCC)nc1C)=O C12(CNC(Nc3ccc(OC)cn3)=S)CCC(CC1)CC2 n1(CCC)ncc(CNC(C2CN(Cc3csc(-c4ccn(C)n4)n3)C2)=O)c1C C1(NC(c2cccc(SCCC)c2)=O)CC2CC(C1)N(C(=O)Cn1cccn1)C2 C(=O)(CCCCC(F)(F)F)NC1(CCNC(c2c(C)nc(C)[nH]2)=O)CCC1 N1(C(C(COC)C)=O)CCC(C2CCN(C(=O)Cc3c(C)nn(C)c3C)CC2)C1 N1(C(C=CC=CC)=O)CC2CCC(C1)N2C(=O)C(C)Oc1ccc(OC)cc1C C1(C(COC)OC)CCCCN1C(=O)NCCCC1(O)CCCC1 c1(C(=O)NC(CC=CC(=O)NCc2cc(COC)on2)(C)C)ncc(F)cn1 C(CCC)(C(=O)NCC1(CNC(=O)CC2C=CCCC2)CCC1)=CCC Cc1ccc(CNC(N2CCCC(n3ccnn3)CC2)=O)c(F)c1F Cc1cccc(O)c1C(=O)NC(C)CN(C)C(C1CC1c1cccs1)=O c1(C(N2CCCC(N(C(C(CC#C)C)=O)C)CC2)=O)cc([N+](=O)[O-])c(C)cc1C Cc1csc2cc(C(=O)NCC(C)CNC(c3csc(=N)[nH]3)=O)[nH]c12 C(=O)(C(CC(F)F)N(C)C(c1cc(OC)ncn1)=O)N1CCC(=CCC)C1 C1(N(C(=O)COc2ccsc2)C)CCCN(C(=O)CCN2CCCS2(=O)=O)C1 c1(C(=O)NC(CC)(CNC(=O)Cc2ccsc2)CC)cc(NC2CC2)ncc1Cl C1(C(N(C)Cc2nc(C)c(C(C)C)s2)=O)CN(CCN2CCCC2)CC1(C)C N1(C(C(C)C(C)(C)C)=O)CCC2CCN(C(=O)Cc3csc(NC4CC4)n3)CC12 C1(C(N2CCC(CC=C)C2)=O)OCC2COCCC12 C1(C(N2CC(CN(C(C3C=C(C)CS3)=O)C)OCC2)=O)CCCC1C1CC1 C1(NC(=O)COC(F)F)CN(C(C2CCN2C2CCCC2)=O)CC2(CC2)C1 C1(CNC(CC2C(C)=NOC2=O)=O)CN(C)CCN1C(=O)CSC1CC1 C(N=c1[nH]c(C(=O)N(CCC(N)=O)C)nc(=N)[nH]1)c1cc(OC)no1 N1(C(CNC(C(COC)O)=O)C)CCN(C(=O)CC2CCCCC2)CC1 CC(F)(F)C(C)(C)C(=O)NC1CC12CCN(C(c1cc(N)nc(Cl)c1)=O)CC2 c1(OC)ccc(I)cc1NC(C1CN(C(c2ocnc2C)=O)CCC1O)=O C1(C(C)(C)C)OCCC1C(=O)NCC=CCNC(=O)Cn1ccc(C2CC2)n1 c1(C(N2CCC(n3cc(-c4n(CC)ncc4)nn3)C2)=O)ccc(P(C)(C)=O)o1 C1(NC(CCCCSC)=O)C(CNC(c2cc(CO)n(C)n2)=O)CCC12CCC2 C(=O)(C(CC)(CC)CC)NCC1C(NC(C(CC=C)c2ccccc2)=O)CC1 C1(CNC(c2c(C)cc(N)cc2)=O)(NC(=O)C2=CCN(C)C2)CCC(F)(F)CC1 N1(CC(Cc2ccccc2)OC)CCC(O)(c2ccc(Br)cc2)CC1 N1(C(C(N2CC(C)C2)C)=O)CC(CNC(=O)CSC2CC2)C(C(F)(F)F)C1 C(=O)(CCP(C)(C)=O)NCC1CCC(C(N2CC(C)C(F)C2)=O)O1 c1(CNC(c2ccoc2Cl)=O)ccc(CNC(c2ccc(F)o2)=O)c(F)c1 C1(C(N(CCNC(c2c(C(=O)OC)c(C)on2)=O)C(C)C)=O)CN(C)CC(C)O1 c1(OC)ccc(C(=O)NCCC(O)CNC(C2CCCN2C)=O)c(N)c1F c1(CNC(c2nc(C(C)OC)oc2)=O)ccc(CN(C)C(C2CC2(Cl)Cl)=O)cc1 C(C(CC(C)C)NC(c1cc(C(F)(F)F)on1)=O)NC(C=CCCC)=O c1(C(=O)NCC2N(C(c3oc(C)c(CO)c3)=O)CC=C2)noc2c1CCCC2 C1(C(=O)NC2C(CNC(=O)COc3ccc(F)cn3)CC2)CCCCC(=O)N1 C1(F)(C(N2C(c3cccnc3)CC(C)C2)=O)CS(=O)(=O)CC12CCC2 C1(C(=O)NCC=C)CCN(C(=O)NCC)C1 C(CNC(=O)Cc1cnsc1)(C(C)C(C)C)NC(c1cnc(COCC)s1)=O C1(S(C)(=O)=O)(C(=O)NC(C2CN(C(=O)CCn3ccnc3)C2)C)CCCC1 CC1CN(C(=O)Cc2ccnc(O)c2)CCC1C(=O)NC(C)C(C)O N1(C(C2CC(C(F)(F)F)(OC)C2)=O)CCN(C(=O)CN(C)C)CC1 c1(CN(C(C2COC(CNC(=O)C(F)OC(F)(F)F)C2)=O)CC)cnn(C)c1 C1(C)(NC(CCc2c(C)nn(C)c2)=O)CCN(C(c2sccc2C(C)C)=O)CC1 Cc1ccc(NC(=O)CC23CCC2CN(C(C2CC(CF)C2)=O)C3)c(C)c1 CC(C)CCCCC(=O)N1C(C(N2Cc3cnn(C)c3C2)=O)CCC1C1CC1 CCC(C)CCC(=O)N(CC(O)CNC(c1sc(Br)nc1C)=O)C c1(OC)c(C(N2CCC(C)N(C(C3CC(=O)N(O)C3)=O)CC2)=O)nc(O)nc1O c1(OC)cc(C(=O)NCC(CNC(=O)C#CC2CC2)C(F)(F)F)ccc1Cl c1(CCC)noc(CCCC(=O)NC(CO)C(C)NC(=O)CC2CC(C)=NO2)n1 C1(C(=O)NCCC2CCN(C(CCOC(CC(C)C)C)=O)C2)CCOC(=O)CC1 c1(OC)c(F)cc(C(=O)NCCN(C(=O)CC2COCCO2)C)c(N)c1F CC1(NC(c2cc[nH]n2)=O)CCN(C(c2ccccc2-c2nc[nH]n2)=O)C1 N1(C(c2c(OC)cccc2CO)=O)CCC(N=c2[nH]nc(C(C)C)o2)(CO)CC1 c1(CN(CC(=O)Nc2cccc(-c3ccno3)c2)C)ccc2ccccc2c1O c1(C(N2CCC(N(C(c3c(OC)c(C)ccc3)=O)C)C2)=O)cc(F)cc(Br)c1Cl CC1CN(C(=O)CCOC2CC2)CC1C(=O)Nc1ccsn1 N1(C(CCc2onc(CSC)n2)=O)CC(NC(=O)C(C)(O)COC)C(C2CC2)C1 c1(CCC(N2C3CN(Cc4ccnc(Br)c4F)CC23)=O)ccc(F)c(Br)c1 C1(CCNC(c2c(C)nc(O)s2)=O)CCCN(C(=O)CSc2n[nH]c(O)n2)CC1 c1(C(=O)NC2CCCN(C(C(CCC)O)=O)C2)cc2ccc(F)cc2nc1O CC(CC(F)(F)F)NC(=O)CC=CC(C)(C)C.C12CC(C1)CN(C)C(=O)C2 S(=O)(=O)(c1ccc(N(C)CCN(C)CCO)cc1Br)NC1C(SC)CCCC1 C1(NC(=O)Cc2ccon2)CCCCCN(C(=O)C(c2cccc(Cl)c2)O)C1 c1(SC)cnc(C(c2nnnn2-c2ccccc2)NCc2ccoc2)s1 c1(C(N2CC(F)CC(NC(CCN(C)CC)=O)C2)=O)c(Cl)ccc(C)c1N C1(C(N(CCCCN(C(=O)Cc2cc[nH]n2)C)C)=O)CCCC(C2CC2)O1 C1(C(=O)NCCCCC(C)NC(C2CCOC2C)=O)CC2(C1)CC2(F)F C1(C(=O)NC23C(CN(C(C(CO)NC(N)=O)=O)C2)C3)C2C3CCC(C3)C12 N1(C(C(C)SCC)=O)CCCC(N(C)C(c2ccc(OC(F)F)cn2)=O)C1 N1(C(c2cnc(CNC(CC3ON=C(C)C3)=O)nc2)=O)CCn2ccnc2C1 C(=O)(C1CSc2ccccc21)NCC1(NC(Cc2nc(NC=O)sc2)=O)CCC1 c1(C(=O)NCC(C)(C)NC(CC2COCC(C)O2)=O)cc(F)cc(F)c1O c1(OC)c(C(N2CCC(O)(C(F)(F)F)C2)C(=O)NC2CCC2)cc(C)cc1C CC1C(NC(=O)CCC2OCCO2)CCCN1C(=O)Cc1cncc(Br)c1 Cc1cc(C)c(NC(=O)C2=CCCN(C(c3csc(Br)c3)=O)C2)c(C)c1 c1(C(=O)NC2CC(C)(C(=O)O)C2)c[nH]c(=NC2CCOCC2)cn1 c1(OC(C)C(=O)NCCCN(C(c2cncs2)=O)C2CC2)ccc2c(c1)CCC2 N1(C(C2CC(SC)C2)=O)CCC2(CCC2NC(c2ccc3c[nH]nc3n2)=O)CC1 c1(C(=O)NC(C2CN(C(C34CCCN(CCC3)C4)=O)C2)C)ccc2cnnn2c1 C1(C)(C(N2CC(CNC(c3ncn(CC)n3)=O)(COC)C2)=O)CCC(=O)N1 Cc1ncc(N)cc1C(=O)NCC(O)CNC(c1oc(Br)nc1C)=O Cc1cc(C(=O)NCC2CN(C(C3CC3c3cccs3)=O)CC2O)cc(C)c1 Cc1cc(N2CC(CN3CCOCC3)C2)nc(=NCC23CCCC2OCC3)[nH]1 c1(C(c2n(C(CC)C)nnn2)NC(C)CSC)ccc(-c2cnco2)cc1 Cc1ncccc1C(=O)NC1CCC1C(=O)NCC1CCCN(C)C1 c1(C(N(CCCNC(=O)C(C)C(C)(C)C)CC)=O)cc(C)c(C)c(S(N)(=O)=O)c1 c1(CNC(C(C)c2cccs2)=O)cccc(C(=O)NCCC2COCCO2)n1 C12(C(=O)NCc3cc(C(=O)NCC4(C(C(C)C)O)CC4)n[nH]3)CC(C#N)(C1)C2 N1(C(Cc2ccc(C)s2)=O)CC(CO)C2(C1)CN(C(C1(F)CCOC1)=O)C2 C1(NC(C(C)SCC)=O)CC(C(=O)N(C)C2CC2)=CC1O C12(C(N3CCC(NC(CC)=O)C3)=O)CCCC1CCN2C(=O)Cc1ccoc1 c1(C(C)=O)cc(C(=O)NCC(C2CC2)NC(c2cc(F)cc(F)c2)=O)c(C)nc1C C1(CCNC(=O)CC2CCC2(F)F)CCN(C(=O)CSC(F)(F)F)CC1 c1(C(=O)NCC(C(C(C)C)C)NC(=O)COC(F)F)ccc2n[nH]cc2c1F N1(C(=O)COCC2CCCCO2)CCCC2(C1)CN(C(c1cnn[nH]1)=O)C2 N1(C(C2(CC(C)C)CC(O)C2)=O)CCC(C)(N2CCCC2)C1 C1(C(N(CC(CC)NC(C2CCOC2)=O)CC)=O)C2CN(C)CC12 N1(C(C(C(=O)OCC)C(C)C)=O)CC2(C1)CN(C(=O)C1=CCCCC1)CC2CO c1(C(CC)C)ccc(C(N2CC(NC(C3CC(C)C3)=O)C(CC3CC3)C2)=O)cc1 C=CC(C(F)(F)F)NC(c1c[nH]nc1CCNC(=O)C=CC1CC1)=O C(=O)(CCN=c1[nH]ccs1)N(CC(CNC(CC1CC(=C)C1)=O)C)C CC1CCCN1CCC(=O)NCCNC(=O)OC1(C)CN(C(=O)C2CC2)C1 C1(CCNC(CC2C(CC)CC2)=O)CCC(C)N(C(=O)C=C(C)C2CC2)C1 C(CCN(C)C(c1cnnc(C)c1)=O)(C(C)(C)C)NC(C(COC)COC)=O CC1CC2CN(C(=O)CC3CCN(C(=O)CC4CC(C(N)=O)=NO4)CC3)CC12 C12(C(=O)NCCC(C)CCNC(=O)C3=CCCC3)CCC(CC1)CO2 Cc1c(NC(C23CC(CNC(=O)CC(F)(F)F)(C2)C3)=O)cccc1Cl c1(C(=O)NC2CC(N(C(=O)CCc3cn(C)nn3)C)C2)ccc(N)c(Cl)n1 C=C(C)CC(C(=O)Nc1cscc1C)NC(=O)Cn1cc(CO)nn1 c1(C(=O)NCC2(CNC(C(CC)F)=O)CC23CCC3)cc(C(=O)OC)sc1C C12(NC(c3cc(C)on3)=O)CCOCC1CN(C(C1CN(C)CCO1)=O)C2 N1(C(c2n(C)ncc2N)=O)C2CCC1CC(NC(=O)CC1COCCO1)C2 c1(C(=O)NCC2(C(F)F)CCN(C(C(OC)OC)=O)C2)cc2ccc(Cl)nc2s1 c1(OCCSC(C)=O)ccccc1F.c1cn(CC(=O)NCC(CO)O)nn1 CCCCCC(CC)C(=O)N1CC(NC(=O)CCCCCCSC)C(O)C1 N1(C(C(C)OCC)=O)CCOCC(NC(C2COCOC2)=O)C1 N1(C(CCC(=O)OC)=O)CCN(C(c2cc(OC)ccc2O)=O)C(CC#N)C1 C1(=CC(C(c2nnc(C)s2)(C)C)=O)Cc2ccc(Cl)cc2C1=O c1(C(=O)NC(CC)CN(C(=O)C(C)(F)C(C)(C)F)CC)ccc2c(c1)CNC2=O Cc1c(F)ccc(C(=O)NC(C)(CNC(=O)C(C)O)CO)c1N Clc1nccc(C(c2nnnn2C2COC2)NC2CC3(C2)CC32CC2)c1Cl N1(C(C=CCCC)=O)CC2CC(C1)C(CO)C2NC(c1sc(CO)nc1C)=O Cc1c(NCC(=O)NC2CCC(C)N2C)ncnc1Nc1ccc(F)c(F)c1 N1(C(C2OCCN(C(C)=O)C2)=O)CC2=C(C1)CN(C(c1nnsc1C)=O)C2 CS(=O)(=O)c1ccc(C(=O)CN2CCC(c3noc(C(F)(F)F)n3)CC2)cc1 S(=O)(=O)(c1cnc2ccc(F)cc2c1)NC1CCC(C(=O)OC(C)(C)C)CC1O c1(CCNC(N2CCC(=CC(=O)Nc3ccccc3)CC2)=O)ccc(F)cc1I C1(C(CO)NC(C2CC(Cl)(Cl)C2)=O)CCN(C(c2cc(C(F)F)ccn2)=O)CC1 C1(CC=C)(NC(c2ccn(CCOC)n2)=O)CCN(C(=O)C(C2CCC2)OC)C1 N1(C(c2c(C)cc(C)s2)=O)CCC2C(C(=O)NCCCC(=O)N(C)C)C2C1 C(CCF)(C(=O)N(C1CCCOC1)C)NC(CCCN(C(C)C)C)=O C1(C(N(C)Cc2cc[nH]n2)=O)CCCCN(C(c2n[nH]cc2Cl)=O)C1 CCCC(CC)CC(=O)N(C1CCN(C(=O)Cn2ccnc2C(C)C)C1)C C=CC(C)(C)CC(=O)NC(CNC(=O)Cc1ccccc1OC)C(C)C(C)C C(=O)(C1=NOC(C)C1)N1C2C(NC(c3c(C)n(CCN(C)C)nc3)=O)C(C2)C1 N1(C(C2(SCC)CC2)=O)CC2(C1)CN(C(=O)C(C1CCC(C)CC1)CC)CCO2 C(=O)(C(F)CCC(C)(C)C)NCCC1CCN(C(C2CC(CCC)C2)=O)C(C)C1 N1(C(C(CC=CC)NC(C2CC(C(C)C)=NO2)=O)=O)CCC12CCCCC2 c1(C(N(C2CCN(C(C3CC(C#C)(O)C3)=O)C2)CC)=O)cccc(N=[N+]=[N-])c1 c1(C(=O)NCCN(CCC)C(C2CCCN(C)C2)=O)cc2n(n1)CCOC2 C12(C(=O)NCCN(C(=O)CC3C=CS(=O)(=O)C3)C3CC3)CCC(CF)(CO1)C2 C1(C(N2C(CC)COCC2)=O)CC(F)(F)CN1C(c1scnc1Cl)=O N1(C(COCCOCCOC)=O)CCC(OCCNC(=O)CCN(C)C)C1C c1(CC2(C(=O)OC3CCS(=O)CC3)CCOCC2)ccc2c(c1)CCO2 S(=O)(=O)(c1ccc(N2CC3CCC(CO)(C3)C2)c(Br)c1)NCCOCOC c1(C(=O)NCC(C)(CC(C)C)NC(C=C(CC)C)=O)sc([N+](=O)[O-])cc1Cl N1(C(C(N)=O)=O)CCn2cnc(-c3cccnc3C(F)(F)F)c2C1 C1(C(=O)NCC2(CCOC)CCC2)(NC(c2cncn2C)=O)CCCC1C N1(C(C(CC(=C)C)NC(=O)C(COC)N(C)C)=O)CC2(COC(=O)N2C)C1 CCC(C#N)(CC)C(=O)N1CCC(C)(NC(=O)CCOc2ccccc2Br)C1 C(c1cccc(CO)c1)=CC(N1C(C(C)(C)NC(c2cc(C)sn2)=O)CCC1)=O C(CC1CCCO1)(C(F)(F)F)NCC1CN(C(C2CCC2)=O)C1 Cn1cc(C(CO)NC(=O)Nc2n[nH]cc2CCC2CC2)cn1 C1(C(=O)Nc2c(C(=O)OCC)scc2)CCCCN1C(=O)Cc1cc(C)n(C)n1 Cc1nn2c(C(=O)NC3CN(C(C4(C#N)CCC4)=O)CC4(CC4)C3)c(C)nc2s1 C1(C(N(CC(CN(C)C(c2sccc2C(N)=O)=O)O)C)=O)(CO)CC1(F)F c1(OC)ccc(Cl)cc1CC(=O)NCC1CC1NC(c1n[nH]c(C)n1)=O N#Cc1cccc(CNC(=O)NC2CC2c2ccc(OC(F)F)cc2)c1 C1(NC(C2N(C(c3n(C)ncc3)=O)CCC2O)=O)CC2CCC(C1)C2O c1(C(N2CC3C(NC(C(C)SC)=O)(C3)C2)=O)sc2cc(F)ccc2c1Cl c1(C(=O)NCC(CC)NC(c2cnn3cnnc3c2)=O)cc(F)c(F)c(Cl)c1F C1(NC(CS(C)(=O)=O)=O)CN(C(C2OCCC2C(F)(F)F)=O)C2CCCC12 C1(C)(NC(c2cc(C)c(C)o2)=O)CCCCC1C(=O)NCCn1cncn1 Cc1cnc(C(N2CC(O)(CN(C)C(c3ccccc3CO)=O)C2)=O)nc1 C1(O)(CNC(CCCOC)=O)CC2CCC(C1)N2C(=O)CCc1cnoc1 c1(N(C(c2cc(C)n(CCN)n2)=O)C)cc(C(F)(F)F)ccc1Br C1(CNC(c2c(-n3c(C)ncc3)nccc2)=O)CCCN(C(=O)C(C)O)CC1 C(=O)(C1=CC(O)C(NC(=O)CCc2nc(O)n[nH]2)C1)N1CC(C)CC(CC)C1 C1(CC(=O)NC(CC(=O)NC)C2CC2)CC(F)CN1C(c1nc(Cl)cs1)=O c1(C(=O)NCC(CCOC)NC(C2C(C=C)C2)=O)[nH]c2ccc(F)cc2c1Cl C1(O)(C(N2CCN(CCNC(C3C(C)(C)C3(C)C)=O)CC2)=O)CCCCCC1 N1(C(C=Cc2n(CC)ccn2)=O)CCOCC(NC(=O)C(C)CC(N)=O)C1 c1(NC(N2CCCCC(CNC(N3CCCC3)=O)C2)=O)cccc2nncn12 Cc1sc(C(=O)NCC2CC(C)N(C(=O)CN3CCOCC3)C2)c(C)c1C CC(CC(=O)NCC(=C1CN(C(=O)CC2CCCC(C)C2)C1)F)CC(C)(C)C C(=O)(C(CNC(=O)C(C)C1CCC1)CC(C)C)N1C(CC(=O)NC)CCCC1 C1(C(=O)N(c2ccsc2)Cc2ccc(Cl)c(Cl)c2)COc2ccccc2O1 c1(C(=O)NCC2N(C(C3CC(C(=O)OC)C3)=O)CC2)cn(C)nc1O c1(SC)ccc(CC(N2CC3CC2C3NC(=O)CN2C(C)CCC2C)=O)cc1 C1(NC(C(C)NC(N)=O)=O)(CNC(=O)CC(C)(F)F)CC2CCC1CC2 C1(NC(Cn2ncn(C)c2=O)=O)CN(C(C2CCCCO2)=O)CC1N=[N+]=[N-] C(=O)(C(C)C(=O)NC1CCCC1C(N1CC(C)=C(C)C1)=O)OC C#CCCC(=O)NC1CCCC1NC(c1cc[nH]c1C1CCCC1)=O C(=O)(C(C)(C)CC(C)C)N1C(C)CCC(NC(C=C(C)I)=O)C1 C1(NC(=O)CC2CS(=O)(=O)C2)CCCN(C(=O)C(F)(F)c2cncs2)CC1 C(=O)(C1=C(C)OCCC1)NC(c1ccc(C)cc1)CNC(C(=Cc1ccco1)C)=O Cc1nc2n(n1)CCN(C(=O)C(C1CCN(C(C3C=CCS3)=O)CC1)C)C2 C1(NC(C(C)(C)F)=O)CC2(NC(=O)Cc3c(Cl)cccc3Cl)COC1C2 CC1OC2(CNc3cc(Cl)ncn3)CC1(NC(=O)CNC(N)=O)C2 CC(C(=O)N1CCN(C(c2csc(=N)[nH]2)=O)CC1c1ccccc1)C(C)(C)C N1(C(=O)OC)CCC(C(=O)NC2CC2CNC(c2c[nH]nc2C(F)(F)F)=O)CC1 Cc1csc(C(=O)NCCc2ccc(CNC(=O)C(C(C)C)N(C)C)cc2)c1Cl c1(N2CCC(C(F)F)(CNC(=O)C3=C(Cl)CCOC3)C2)ccc(F)cc1[N+](=O)[O-] CN1CC(C(=O)NC2CC(C(=O)NC(C)(C)C)C2)C(C(F)(F)F)C1 Clc1cccc(CNC(=NCC2CCOC2)NCC23CC(CO2)C3)c1 C1(CNC(c2c(C)ncs2)=O)CN(C(=O)C(C)CC(C)C)CCC12CCOCC2 c1(CC(N2CC(C(C)NC(C(CC=CCC)C)=O)C2)=O)ccc(F)c(F)c1 c1(CC(=O)N(C(CCNC(CC=C)=O)C)C)cn2cc(C)sc2n1 C#CC1(O)CC(C(=O)NC2CC(CNC(=O)CC(C)CC)C2)C1 O=Cc1cccnc1-c1ccc(CN(CCO)CCO)s1 C(=O)(C1=C(F)CN(C(c2ccc(C#N)o2)=O)CC1)N(CC(O)C1CC1)C C(=O)(C(F)C(F)(F)F)NC(CNC(C(CC)c1ccccc1)=O)(CC)CC N1(C(C2N(C(C(CC)n3ccnc3)=O)CC2)=O)CCOCC1CN(C)C C1(OC)CC(CNC(c2cc[n+]([O-])cc2)=O)N(C(=O)C(C)Oc2cccnc2)C1 O=C1NC(=O)C(CCNC(c2ccc(CO)s2)=O)N1 C1(NC(C=CC(=O)OCC)=O)CCC(C)N(C(c2ccc(C(C)C)o2)=O)C1 N1(C(CC(C)CF)=O)CCOC2(CCCN(C(c3cc4n(n3)CCO4)=O)C2)C1 c1(C(N2C(CNC(=O)CN3CCCCC3)CCC2)=O)cccc2c1OCC(=O)N2 c1(C(=O)NC2CCN(C(=O)Cn3cccc3)C23CCC3)ccc2ccccc2n1 c1(-n2cc(CCNC(CC)=O)nn2)cccc(O)c1F C1(C2(O)CCC(=O)CC2)(C(=O)Nc2ccc(-c3nc(C)on3)cc2)CC1 c1(C(=O)Nc2ccc(C#N)s2)ccc2c(C(=O)N=c3cncc(Br)[nH]3)n[nH]c2c1 N1(C(C(COC(C)=O)C)=O)CC=CC(C(=O)NCCc2cnn(C)c2)C1 C1(OC)CC(CCNC(c2csc(F)c2)=O)N(C(=O)C(CC2CCCO2)OC)C1 C(=O)(N1CC(O)CCO1)C1CCN(C(C2CC2(F)F)=O)CC1 C(N=c1ccnc(Cl)[nH]1)C1C(C)CCN(C(=O)CNC(=O)CC(F)(F)F)C1 CN=C(NCCN1CCCC1)N1CCC(CSc2ccc(C#N)cc2)C1 C12(C(=O)NC3CC(NC(C4CC4C(F)F)=O)C3)CC3CC(C(=O)N1)C2C3 C1(C(=O)NC(COCC)C(=O)NC2CC(C)(O)C2)CC2OC1C1CC21 N1(C(C2(OC)CC2)=O)CC(C(=O)O)C2(C1)CN(C(c1cc(O)c(Br)c(O)c1)=O)C2 c1(C(C)C)nn(C)cc1C(N1CCCC1(C)CNC(=O)Cc1cn[nH]c1)=O Cc1c(C(N2CCCC2CCCNC(=O)C(F)C(C)C)=O)sc2ccc(Cl)cc12 c1(OC)cccc(N2CC(NC(=O)CC3CCC(F)(F)C3)C(C)(C)C2)c1[N+](=O)[O-] c1(C(=O)Nc2cn(COC)nc2)ncccc1Oc1cccc(C)c1 c1(C(N2C(C)C(C)N(C(=O)CC(C)C(F)(F)F)CC2)=O)ccc2c(c1)COCC2 C1(O)(CNC(CCC2CCN(C(c3c(CC)n(C)cc3)=O)C2)=O)CCC(C)(C)C1 Cc1c(C(=O)NCCCOCCN(C)C(C2CCS(=O)(=O)N2)=O)cnn1C N1(C(C(=Cc2cnc[nH]2)C)=O)CCN(C(C2C3CCC(=O)C23)=O)CC12CC2 C(=O)(C1CCc2nccn21)N1CC(CS(C)(=O)=O)N(C(c2cnco2)=O)CC1 C12(C(=O)NCCC3N(C(c4cn(C(C)C)nc4)=O)CCC3)CC3CC1C2C3 C1(C(N(C)Cc2ncccn2)=O)CCC(C2CC2)N1C(C1CC(C)(O)C1)=O c1(C(N(C(CCNC(c2cc(C)no2)=O)C)C)=O)sc(N(C)C)nc1C c1(N(C)CCNS(=O)(=O)CC2CC(O)CN2C)ccccc1Cl n1(C(C)(C)C)cc(Br)c(C(N2CCN(C(c3ccnnc3O)=O)CC2)=O)n1 C12(CNC(C(CNC(=O)C(F)=CC3CC3)OC)=O)CCC(CC1)C2 C1(CNC(CN(C)C2CC2)=O)(NC(=O)CC2CC23CC3)CC2CCC1CC2 CCCC(C(=O)NC1(CCNC(=O)C(C)OCC)CCCC1)NC(N)=O C(=O)(C(CNC(=O)Cn1cc(Cl)cn1)CC(C)C)N1CCC(C)(CC)C1 N1(C(C2N(C(C)=O)CCC2)=O)CCN(C(C2C(C(=O)OC)C2(C)C)=O)CC1CF N1(C(C(C)n2cccn2)=O)CCN(C(c2ccccc2)=O)CC(C)(F)C1 S(=O)(=O)(c1ccc2c(c1)CC(=O)N2C)N1CCCC(C)(C(=O)NCC(=O)OC)C1 N1(C(COCCC)=O)CCN(CC(=O)NCC2(O)CC2)CC1 c1(CC)ccc(C(=O)N(C)CCN(C(=O)Cc2ccno2)C)cc1CC C1(NC(c2cccnc2)=O)CCC2(CCNC2)CC1 C=CC(C)(O)C(=O)N1CCC(c2cc(CNC(C3CC3(C)C)=O)on2)CC1 CN1N=C(C(=O)NC2CCCC2CC(=O)NC2CC23CCCCC3)CCC1=O C1(C(N2CCC(OCC(=O)NC(c3ncccn3)C)C2)=O)CC(=O)NC(=O)N1 c1(C(=O)NCCC2CC(NC(CCc3cc(C)no3)=O)C2)cc(C)nn1C c1(-c2cn(-c3c(C(=O)NC4C(C)CC4)cccc3)nn2)ccc2c(c1)OCCO2 CCCN=C(NCCc1cccc(C(=O)NC)c1)N1CCC(C2CCCC2)C1 C1(NC(CCOC)=O)CCN(C(c2c(S(C)(=O)=O)cnn2C)=O)CC(C)(C)C1 c1(-c2cc(OC)ncc2F)ncn2c1CN(Cc1ccc(Br)cc1O)CC2 c1(OC)ccc(NC(=O)CC(C(C)C)NC(C2(N(C)C)CCC2)=O)cc1C c1(OCCOC)cc(O)ccc1NC(=O)NC(Cc1ccccc1)C(=O)OC O=C(CCCCCCBr)NCC1CCC(C(=O)NCc2ccc(F)cc2)CC1 C1(C(=O)NC2CC3CC2N(C(C2CC4(CCC4)CO2)=O)C3)Cc2ccncc2N1 c1(CC)cc(C(=O)Nc2ccccc2CO)n(C)n1 c1(C(N(C2CCN(C(c3noc4c3COCC4)=O)C2)C)=O)ccn2cnnc2c1 c1(COC)cccc(C(=O)NC(C)C(C)NC(C2CCCC2O)=O)c1 c1(C(N2CC(OCCNC(=O)CC3CC(=O)NC3=O)C2)=O)ccc2c(c1)CCO2 CCC(C)C(C)C(=O)NCC1CN(C(=O)C=CCCc2ccccc2)CCO1 CC(C)CC(CNC(=O)C(C)Nc1ccccn1)NC(=O)CN1CCC1C Cc1cc(C(N2CCCCC2CN(C)C(C23CC(CF)(CO2)C3)=O)=O)nc(C)c1 N1(C(=O)COCCF)CCC2(CCCN2C(c2[nH]cc3c2CCCC3)=O)C1 CCCCC(C(=O)N1CC(N(C)C(c2c[nH]c(-c3ccncc3)n2)=O)C1)C(C)C c1(C(=O)NC(CN(C(c2cn(CC=C)nn2)=O)C)C)cc(C(N)=O)ccc1C n1(CC)ncc(C(=O)NCC2CCN2C(c2cnc(SC)s2)=O)c1Br CC1(C)CCC(NC(=O)Cc2ccno2)C(CNC(c2ccc(Cl)nc2N)=O)C1 C1(NC(C2C(OC)CC2)=O)CC2CCC1N2C(c1cscc1Br)=O c1(SC)ccc(C(N2CC(N(C)C(C3CCCOC3C)=O)C2)=O)cc1Br C(=O)(CCC(CC)CC)NC1C(C2CCN(C(C=CC=CC)=O)CC2)OCCC1 O=C(C(CC(F)(F)F)c1ccc(F)cc1)NC1CCC1NC(=O)C1=CCCOC1 CC(CN(C)C)CCC(=O)N(CC(C)(C)CNC(C1(CN(C)C)CC1)=O)C C1(NC(COCCCC)=O)CCC2CC1CN2C(c1cncc(C(F)(F)F)n1)=O N1(C(c2ccc(CC(C)C)s2)=O)C2CCC1C(CNC(C1CCC1)=O)C2 N1(C(C(n2c(C)ccn2)C)=O)CC2CCC2(NC(=O)CCCc2ccsc2)C1 CC#CCCCC(=O)NCCN(C(=O)CN(C)CCOC)C(C)C CCC(C)(O)C(=O)N1CCC(C(C)(C)NC(C2CN(S(=O)(=O)CC)C2)=O)CC1 C1(C(=O)NC2CCCC(NC(C3(C)CC3)=O)C2)COc2cc(Cl)ccc2O1 N1(C(C(CC)Cc2cccc(C)c2)=O)CC2CC(C1)C2NC(=O)CSC(F)(F)F C(=O)(CC(C)CNC(=O)CC(C)F)NC(CC)CO c1(-n2cc(-c3c(C)ocn3)nn2)cccc(NC(=O)COc2ccccc2F)c1 CN1N=C(CC(=O)NCC=CCNC(C2CNC(=O)N2)=O)CC1=O c1(OCC)ccc(OC)cc1NC(=O)Nc1c[nH]c(C(=O)NC)c1 CCCC(O)CC(=O)N(CCCNC(=O)CC1CCCCC1(F)F)CC N1(C(=O)NC)CC(C(=O)NC2CCC2CNC(=O)C(C)C2CCCC2)C1 Cc1sc2ncc(C(=O)NC3(CCNC(C45CC6CC4C5C6)=O)CCC3)n2c1C N1(CC)CCC2(CCN(C(=O)CC(C)C3CC3)C2)C1 C1(C(=O)NCC(c2ccc(F)cc2)NC(c2cc(C(C)=O)on2)=O)CC2C=CC1O2 CC1CC(C(=O)NC2CC2)CN(C(=O)CC2CC23CC3)C1.C1(=O)CN1 c1(C(=O)NCCC(C)NC(CCC2C(C)=NNC2=O)=O)ccc2ncsc2c1 C=C(C)C(C)(C)C(=O)NCC(C)(C)CCNC(C1CCN(C2CCSC2)CC1)=O CC(C(=O)NCCN(C)C(C1(n2cc(C#N)cn2)CC1)=O)C(C)S(C)(=O)=O CN1CCN(C(C2CC(O)C2)=O)CC1C(N1CC2CCC2C1)=O C1(C(=O)NC2C(=O)NOC2)CC2(CCN(C(=O)C(F)(F)c3ccco3)CC2)CO1 N1(C(C=CS(C)=O)=O)CCC2(CCN(C(c3ccnn3C(C)(C)C)=O)C2)C1 Cc1cc2scc(CCNC(=O)COc3ccccc3)c2s1 C1(CC=C)(NC(=O)C=CC(C)(C)C)CCCN(C(=O)CCc2ccc(C)cc2)C1 N1(C(c2c(C)csc2)=O)CC(CNC(c2[nH]nnc2C2CC2)=O)OC(C)(C)C1 c1(CC(=O)NCCNC(C2CN(C)C(=O)C2)=O)c[nH]c2ccc([N+](=O)[O-])cc12 C1(CC(=O)NCC2(C(=O)NCC(CN(C)C)(C)O)CC(F)C2)CCC(=O)C1C C12(C(N3CC4(CN(C(C(C)SC)=O)C4)C3)=O)CCC(=O)N1c1ccccc1S2 N1(C(CCC=C)=O)CC(NC(=O)Cc2ccccc2C)C(C2CC2)C1 c1(C2C(C(=O)NC(c3n(C)ncc3)(C)C)C2)cc2ccccc2o1 N1(C(c2ccc(C)cc2Cl)=O)CCC2(NC(=O)CCOCC3CC3)CCCCC12 c1(C(=O)NC2(CO)CN(C(C(C=C)(C)CC)=O)C2)nc(O)nc(O)c1F C1(CNC(C2CC2(Cl)Cl)=O)CCN(C(C23CCCCC2C3)=O)CC1 c1(CN(C(CCC(=C)C)=O)CC)cc(C(F)(F)F)cc(F)c1 C(=O)(C#CC1CCCCC1)NC(C)CCN(C)C(c1cc(C#N)ccc1Br)=O c1(CN2CC3C(C(N4CC(N5CCC5)C(O)C4)=O)C3C2)c[nH]c2ccc(Br)cc12 c1(C(=O)NCC(=C)CCNC(=O)C(C(C)C)OCC)ccc(S(N)(=O)=O)o1 c1(OC)ccc2nc(C(=O)NCCCNC(=O)CCN3CCC(O)CC3)cn2n1 c1(C(N)=O)ncn2c1NC(=O)C(CC(=O)NCCc1ccc(C)c(Br)c1)C2 C1(CC(N2CC(C(N)=O)(CNC(C(C)CC3CCC3)=O)C2)=O)SC(=N)NC1=O c1(C(=O)OC)c(NC(C2CC(C(=O)Nc3cc(O)nc(Cl)c3)C2)=O)cccc1F c1(N2CC3CCS(=O)(=O)N3CC2)[nH]c(=NCC2CSC2)nc2scnc12 c1(CC)cnccc1C(=O)N(C)CC1(O)CCN(C(C2CC2F)=O)C1 C(=O)(C(CC(C)C)N(C)C)N1CC(CCNC(c2c(CC)nns2)=O)OCC1 c1(OC)ccccc1CC(C)=CC(=O)NCC1CCCCN1C(=O)CC(C)(C)O CCC(C)CCC(=O)N1CC(NC(c2ccc(C)c(OC)c2)=O)C(O)C1 Cc1nccc(C(=O)NCC(C)CNC(C23CC(C)C2C3)=O)c1N C1(C(N2CC(C(=O)N(C)Cc3ccnn3C)(SC)C2)=O)CC2(CCC2)C1 NC(C(=O)N(CCC1CC1)C1CC1)c1cscn1 N1(c2cc(NCC3CCC(C)(C)CO3)nc(C)n2)CCC2(CC(=O)N(C)C2)C1 c1(CNC(C(c2nocc2C)N(CCCC#C)C)=O)cccc(Br)c1 N1(CC(N2C3CN(C(C(C(CC)O)C)=O)C(CC3)C2)=O)Cc2ccccc2C1=O CC1CN(C(c2cn(C3CC3)nn2)=O)CC(C)N(C(c2ccc(=N)[nH]c2Cl)=O)C1 c1(C(=O)NCCC2(C(=O)OCC)CCC2)ccc2c(c1)CN(C)S(=O)(=O)N2C C1(C(C)NC(Cc2ncc(C)o2)=O)CCCN(C(=O)Cn2cnnc2)C1 C12(NC(C3(CC)CCN(C(=O)C=Cc4cc(C)no4)C3)=O)CCCN(CCC1)C2 Cc1cc(C(=O)N(CCNC(=O)C=CCF)Cc2ccccc2)no1 Cc1nc(C(=O)NCC(C2CC2)NC(C23CCCC2C3)=O)nn1-c1ccccc1 CC1CN(C(c2cnn3c2SCC3)=O)CCC1CNC(=O)COC1CC=CC1 C(=O)(CCC1=CCc2ccccc21)NC(C1OCCN(C(CC)=O)C1)C Cc1ccc(-c2nc(CC(=O)NC34CC(CNC(c5ccon5)=O)(C3)C4)cs2)o1 C1(C(N(CC(C)(C)CNC(=O)CS(=O)(=O)NC)CC)=O)CCCC(F)(F)CC1 N1(CC(=O)NCCC(=C)CNC(=O)CC(C)CC(C)C)CCSC2CCCCC12 c1(CC)noc2ncc(C(N3CCCC3C(C)NC(c3cncnc3)=O)=O)cc12 N1(C(CC=C(C)C)=O)CCC2(CC1)OCCCC2NC(=O)CC1=NNC(=O)C1 C(=O)(CC1=CCN(C)CC1)N1CC=CC(NC(c2ccn(COC)n2)=O)C1 c1(C(=O)NCC(CNC(=O)C(=Cc2c[nH]cn2)F)OC)ccnc2[nH]cnc12 CC1CC(F)(F)CN1C(=O)CCN(C)C(C1CCC(C)(C)C1)=O C1(NC(=O)C2=CCCC2)CS(=O)(=O)CC1NC(C1(CCF)CCOCC1)=O CCCC(C(O)C(=O)NC(CC)CC(=O)OC)NC(C1C(C)C1C)=O c1(CCC(=O)NCCN(CCC)C(=O)C2CC2)ccc(OC(F)F)cc1 CC1CN(C(=O)C(c2ccc(Cl)s2)=O)CC(c2ccccc2)O1 Cc1cccc2nc(CCNC3CC3(C)C3(C)CC3)cn12 CC(C)CC(C)C(C)Nc1ccc(C(F)(F)F)nc1OC(C)C c1(N(C)CC2CSc3ccccc3O2)nc(=NCC(C)(C)F)[nH]c2c1COC2 c1(OC)ccc2cc(C(=O)NCC(CO)NC(C34CC(OC)C3C4)=O)ccc2n1 c1(NC(CC2CC(NC(C(C(=O)OC)C)=O)C2)=O)cc(C(C)=O)ccc1Cl Cc1c(CN2C(CNOC(c3ccc(Cl)cc3Br)=O)CCC2)oc2ccccc12 Cc1cnccc1C(=O)NC1CC(CNC(=O)CC(C)(C)C2CCCCC2)C1 c1(CS(=O)(=O)N(C2(C)C3COCC23)N(C(C)(C)C)CCO)ccccc1N C(=O)(C1CCc2cc(Br)ccc21)NCCCCCC1CCN(C(C)=O)CC1 C1(C(C)C(=O)NCC2(CN=[N+]=[N-])CC2)CCCN(C(=O)Cc2cn(C)cn2)C1 c1(CNC(CCn2cc(-c3ccc(C(=O)O)cc3)nn2)=O)ncc(F)cc1F C1(O)(CN(C(C(COCC)C)=O)C)CCCN(C(=O)Cc2cccc(F)c2)C1 c1(CC(N2CCC(NC(C(C)CO)=O)C2C2CC2)=O)ccc2c(c1)CC2 c1(CC)[nH]nc(C(=O)NC(CCN(C)C(c2n[nH]cc2Cl)=O)C(C)C)c1C Cc1nnc2n1CC(C(=O)NCC1C=CC(NC(c3ccc(Br)o3)=O)C1)CC2 C12(C(N3C(CNC(CC(N4CCCCC4=O)C)=O)CC3)=O)CC(C1)C(C)O2 CC1CCOC(C(=O)N(C)CC2CCN(C(=O)CC3CNC(=O)O3)CC2)C1 c1(C(N2CCCC(C)(C)C2)C(=O)NCCOC2CC2)cccn2ccnc12 C(=O)(CC(C)(C)CC(=O)NC1CCCCN(C(c2n[nH]c(C)c2F)=O)C1)OC n1(C(CC)C)ccc(=NC(=O)C2CC(NC(=O)CN=[N+]=[N-])C2)[nH]1 c1(C(=O)NC2CC(NC(c3ncc(C#N)cc3Br)=O)C2)cc2ccnc(Cl)c2[nH]1 Cc1cnccc1C(N1CC(NC(=O)C=CC2CCC2)C(c2ccccc2)C1)=O C1(NC(c2c(C)cc(C)s2)=O)CC2CN(C(c3ccc(F)c(C)c3)=O)CC2C1 C1(CNC(C(CC)SC)=O)(OC)CCN(C(C2CC(n3cnnc3)C2)=O)C1 c1(OC)cc(F)c(F)cc1C.C12CCC3CC13CNC(=O)N2 C1(OCC)CC(N=c2[nH]c(=NCC3(C)CCN(C)C3)[nH]c3c2CCCC3)C1 CC1(C)C=C(C(=O)NCC2(C)CCN(C(=O)C(N3CCOCC3)C3CC3)C2)C1 c1(OC)cnnc(C(=O)NC2CCC(CC(=O)NCC(C)(C3CC3)OC)CC2)c1 c1(C(=O)NCCC2(O)CN(C(c3cn4c(n3)SCC4)=O)C2)ccc(O)c(CO)c1 C1(NC(C2C(C(=O)OC)C2)=O)CC2CCC(C1)N2C(c1cc(F)c[nH]1)=O C1(O)(CNC(C(n2cc(Cl)cn2)C)=O)CN(C(=O)C(C2CC2)Sc2ccccc2)C1 C(CCC(C)(C)C)(C(N)=O)NC(C(=O)Nc1cnc(CC)nc1C)C c1(C(=O)NC2COCC2NC(C2CSCCS2)=O)ccc2nnc(O)n2c1 Cn1cnc2c(NC(C)(C)C)[nH]c(=NC3CN(CC4CC(O)C4)C3)nc12 C(C1CCCC1)=CC(=O)NC1(CC(=O)NCCc2nncs2)CCC1 c1(C(N2CC3(CN(C(C4CCC(N=[N+]=[N-])C4)=O)C3)C2)=O)cc(F)c(O)c(Cl)c1 c1(C(C(N2CCC(C(C)NC(c3c(C)cnn3C)=O)C2)=O)=O)ccc(F)c(F)c1 C1(C(=O)NCCOCCCCC)CCN(C(C23CCC(OC)C2C3)=O)CC1O C1(=CCNC(C(CC)c2ccccc2)=O)CCN(C(C2CC(C(F)F)C2)=O)CC1 Clc1nonc1CN1CCCC1C1CCC1 N1(C(CCCCC#N)=O)CCCC(F)(CNC(=O)C2=C(Cl)CCCC2)CC1 C1(CC(N2CC(NC(c3ccsn3)=O)C(C(F)F)C2)=O)CC2(CCC2)CCO1 C(=O)(C(C#N)C(C)(C)C)N(C)CC1CCCCN1C(=O)CC1CCCC1 CCCC(C)(C)C(=O)NCCC12CCC(C1)N(C(=O)C(O)CN(C)C)C2 N1(C(C(c2ccccn2)C)=O)CC(F)CC1CNC(C1CCC=CO1)=O C(=O)(CCCCCC(C)(C)C)NC1(C2CCN(C(C=CC(C)(C)SC)=O)C2)CC1 N1(C(CCOC(C)=O)=O)CCC2CCC(NC(=O)Cc3cc[nH]n3)C1C2 CC1CC(C(N2C3CCC(C3)C2CNC(=O)Cc2nc[nH]n2)=O)CC(C)(C)C1 c1(C(C)(C(=O)O)NC(C(C2CCCCC2)C)=O)ccc(NC(=O)OC(C)(C)C)cc1 C(=O)(C(CCCO)c1ccccc1)N1CCC(N(C)CCO)CC1 N1(C(C(C)=CC2CC2)=O)CCCC(O)(CNC(=O)CN(C)C(N)=O)CC1 Cc1nc(C2CC2)sc1S(=O)(=O)N1CCN(C2CC(C)CC(C)(C)C2)CC1 c1(C(N(CCC)CCNC(=O)CCOCC(F)F)C)cn(-c2ccccc2)nn1 C1(F)(CNC(c2cnn(C)n2)=O)CCN(C(=O)CCSC(F)(F)F)C1 C(=O)(CC(C)CC(F)(F)F)NCC1C(C)(C)CCN(C(c2n(CC)nnc2)=O)C1 C(=O)(C(C(C)(C)CC)OC)N(CC(C)NC(=O)CCc1cc(Cl)no1)CC C(=O)(CN=S(C)(C)=O)N(CCNC(=O)Cc1cnsc1)CC C1(C(N2CC(NC(c3cc4sccc4cn3)=O)C(O)C2)=O)CC2(C1)CC(F)(F)C2 N1(C(c2ccc(N)c(F)c2)=O)CCCC12CCN(C(=O)C#CC1CCCOC1)C2 c1(OC)cnc(Cl)cc1C(=O)NCCCC1CCCN1C(=O)C(C)C(C)C N1(C(C2(COC)CN(C(C(CC)NC(N)=O)=O)C2)=O)CCC2CC12C c1(OC)ccc2[nH]c(C(=O)NCC3(NC(=O)C(F)OC(C)=O)COC3)cc2c1OC Cc1nn(C)c2ccc(C(=O)NCC3(F)CCC(CNC(=O)CC(C)F)C3)cc12 C1(C(=O)NC(C)CCCNC(C23COCC(C2)C3)=O)CCN(CCO)C(=O)C1 C(C(C)(COCc1cn(CC2C3CCCC23)nn1)Cn1cccn1)OC C1(CNC(C2CC(n3ccnc3)C2)=O)CC2CC2N1C(C1CC(F)(F)C1)=O Fc1ccc(F)c2c1CCN(C(=NCCOCC(F)(F)F)NCC1CCCO1)C2 C1(CCC)CN(C(c2cc(CC)ccn2)=O)CC1NC(c1ccc(SC)nc1)=O C1(C(N(C(C)C(N2CC(C)(O)C2)=O)C2CC2)=O)CC2CCC(C1)C2 c1(C(N2CCC(C(CNC(CS(C)(=O)=O)=O)F)CC2)=O)ccnc2ccsc12 C(c1ccc(C)cc1C)=CC(=O)NC1CN(C(COC(CC)C)=O)CC1F S(=O)(=O)(c1cccc(=NC2CCN(S(C)(=O)=O)C2)[nH]1)N1CCCC(C=C)C1 C(=O)(C(C)(C)CS(C)(=O)=O)NC1C2CN(C(CN3C(C)CC3)=O)CC1CC2 C12(CC(=O)NC3C(C)CN(C(C4(F)CC=CC4)=O)C3)CC3CC(CC(C3)C1)C2 c1(C(=O)NCCN2C(CCCC)CCC2)cc(F)cc([N+](=O)[O-])c1N CC1OC2(C)CC1(NC(=O)C(C)NC(c1ccccc1)=O)C2 N1(C(c2cnc(C(C)C)[nH]2)=O)CCC(NC(=O)CCC2(C)CC2)C(CO)C1 C1(CC)(NC(C2CC2F)=O)CCCN(C(=O)CC=Cc2ccc(C(C)C)cc2)C1 C1(C(=O)NCCC2CCN(C(C3(CCOC)CC3)=O)C2)CCCC12CC2 C1(C)(C(=O)NCCCC(C)NC(=O)Cc2ccc(F)cn2)CC=CCC1 N#Cc1ccc2c(CN3CC4C(C(=O)NC(c5ccccc5)CO)C4C3)c[nH]c2c1 c1(C(=O)NCCC(CNC(Cn2nnc(C)n2)=O)O)ccc(C(N)=O)nc1 C(C)(C(C(=O)N1CCNC(=O)C1)NC(=O)C(CSC)OC)OC Cc1cccc(CNC(=O)CCC2CCN(C(C3(C)CC(C)(C)C3)=O)CC2)c1C N#Cc1ccc2c(c1)CCN2C(=O)C(C1CCC1)NC(=O)C=C1CCOCC1 C1(NC(CC2N(C(C)C)CCC2)=O)CN(C(=O)Cc2cnsc2)CCC12CCC2 n1(CC)cc(CNC2CCN(Cc3c(Br)cncc3Br)CC2)c2cccnc12 C1(NC(CC2(C=C)CC2)=O)COC2(C1)CN(C(c1ccc(-c3cc[nH]n3)s1)=O)C2 Cc1ccc(C(N2CC(NC(c3coc(C(F)(F)F)n3)=O)C3(CC3)C2)=O)c(Cl)c1 Cc1cccc2[nH]cc(CC(=O)NC3CCCN(C(=O)Cc4cnsc4)C3C)c12 N1(C(CN(S(CC)(=O)=O)C)=O)CC(C)CN(C(c2cn(C)nc2OC)=O)CC1C C(CC(C(=O)N1CCC(CNC(=O)C(C)SC(C)C)CC1)OC(=N)O)OC c1(-c2cc(C(N(CCC(C)NC(=O)C(C)CF)C)=O)n[nH]2)ccccc1Cl c12cc(ncn1)N1CCCC1CCC(=O)NC2.c1(OCC(=O)OC)ccccc1 c1(C(N2C(CN(C(C3C(C)C3)=O)C3CC3)CCC2)=O)cc2cccnc2o1 c1(C(=O)NC(C)C(C)NC(=O)Cn2cnc(C(F)(F)F)n2)ccc(C(F)F)cc1 C1(O)(C(=O)OC)CN(C(=O)C(C2CCCO2)NC(=O)C(O)CN2CCCC2)C1 C1(NC(CCOCCOC)=O)CC(OC)CN(C(c2nnn(C)c2C)=O)C1 C=C(C)C(C)(O)C(=O)N1CC(C(C)(C)O)(CNC(=O)Cc2c(Cl)cnn2C)C1 c1(C(=O)NC2(CNC(=O)COC3CCC3)CCOC2)cnn2ncccc12 C(=O)(CS(C)(=O)=O)N1CCC(N(C(c2c(CC)nco2)=O)CC)C1 C1(NC(C(C)(C2CCC2)NC(c2ccc(Cl)cn2)=O)=O)CC(=O)NC(=O)C1 C1(CCNC(c2cc(Cl)c[nH]2)=O)CN(C(c2ocnc2C2CC2)=O)CCCO1 C1(C2CCCN(C(c3nnn(C(C)C)c3C)=O)C2)(NC(C(CC=CC)C)=O)CC1 c1(C(N2CCC3CCC(NC(C4CCC4)=O)C2C3)=O)ccc2cc(O)ccc2n1 N1(C(c2cc(CC)[nH]n2)=O)CC(C)(C(N2CCCC(CN=[N+]=[N-])C2)=O)CC1(C)C N1(C(C(CC)(F)F)=O)CCC(C)C(NC(c2cc(Cl)ccc2Cl)=O)C1 C1(C(=O)O)C2C=CC(C2)C1NC(=O)C(c1ccc(F)c(Cl)c1)O c1(C(=O)NCC2CC(NC(CC(=O)NC)=O)C2)cc(C(C)C)nn1C CC1CCC(C)N1C(C)C(=O)NC1(CF)CCN(C(c2csc(=N)[nH]2)=O)C1 c1(C(OP(C)(=O)COCCn2cc(C(C)(C)CC(=O)OC)nn2)C)ccc(Br)cc1 Cc1csc2cc(C(=O)N(C3CCC(NC(=O)C(=O)N(C)C)CC3)C)[nH]c12 Cc1cc(C(N2CC(C)C(Nc3nccnc3C#N)C(C)C2)=O)c(F)cc1F C1(NC(CCC(C)NC(C=CC(C)C)=O)=O)CCCCNC1=O C1(NC(C(C)OCCOC)=O)CCCCC1N(C(=O)C(=Cc1ccccc1)C)C c1(N2CCCC(CCC)CC2)cc(Br)ccc1S(=O)(=O)NCC1CC1 C(=O)(C(C)(C)S(C)(=O)=O)NC1CC(CNC(c2ccc(OC)c(C)c2)=O)CC1O S(=O)(=O)(c1ccc(Br)cc1NCCn1ncccc1=O)N1CCC(C#N)C1 N(C1CCCn2ccnc21)C(CC(C)CNC(=O)C(C)(C)C(F)F)=O c1(Cc2cc(C(C(=O)Nc3ccc(F)cc3)N(C)CC)on2)ccc(F)cc1F C1(O)(C(C)NC(C(C)OCC2CC2)=O)CCN(C(c2ccc(C(F)(F)F)[nH]2)=O)C1 C1(O)(CNC(=O)CCOC2CC2)CCN(C(c2cn(CC3CCOC3)nn2)=O)C1 N1(C(c2cc(C)sn2)=O)CC2(CCCC2NC(c2cncn(C)c2=O)=O)C1 c1(OC)ccc(-c2ccc(NC(c3ccc(I)c(Br)c3)=O)nc2C)cc1C(C)C CCC(COC)C(=O)NC(C)CCC(=O)NC(C)COCC1CC1 CC(C(=O)N1CC(F)CC1CNC(C1(c2cncs2)CC1)=O)C(F)F CCCC(C(O)C(=O)N1CC2CC1CO2)NC(=O)CCCn1cncn1 c1(NC(C23CC2CN(Cc2ccc(Cl)nn2)C3)=O)ccc(F)c(Br)c1 C#Cc1cncc(C(N2CCCC(CNC(C3CS(=O)(=O)C3)=O)C2)=O)c1 CCCC(F)C(=O)N1CC(O)(c2cn(-c3cccnc3F)nn2)C1 CC(C)(C)C(O)C(=O)NC1CCN(C(c2ccc(CN3CCCC3)cc2)=O)C1 CCC(C)C(C)(c1nnnn1C1CC1)Nc1cncnc1CC c1(C(=O)Nc2cc(C)c(Oc3ccccc3)cc2)c(Cl)ccc(Br)c1F N1(C(c2c(CC)[nH]cc2)=O)CCC2(CC1)CC2NC(C1(C)CNC(=O)C1)=O c1(C(C(=O)N(CCN(C(=O)C=CC(=O)NC2CCOCC2)C)C)O)cncn1C c1(C(N2CCN(CCN(C(C(C(C)SC)O)=O)C)CC2)=O)cnc2[nH]cnc2c1 Cc1cnncc1C(N1CC2C(NC(C3(c4ccccc4F)CC3)=O)C2C1)=O n1(CCCC)cc(C(=O)NCC2CCCN2CC(=O)Nc2nccs2)c(C)n1 C#Cc1ccc(C(=O)N(C(C)C(=O)NCCc2nnc(O)n2C)CC)cn1 C1(CNC(C(C2CCOC2)OC)=O)CCN(C(C23CCC(C)(C2)OC3)=O)CC1C C1(O)(C(C)CNC(=O)C(N)=O)CCN(C(c2cnc(C(C)(F)F)s2)=O)C1 N1(C(CNC(C(C)C#N)=O)=O)CC(O)CC(C)(C)C1 N1(C(CC2CCC(=O)N2)=O)CCC2CCC(C1)N2C(C1Cc2ccccc2CN1)=O CC1CN(C(=O)C=CC(=O)NC2CC2)CC(C)N(C(c2cncc(Br)c2)=O)C1 N1(C(C(COC)C)=O)CCCC(CNC(c2csc(Cl)c2)=O)C1 c1(C(=O)NCC2CCC(NC(c3cnsn3)=O)C2)nsc2c(Cl)cccc12 CC(C)C(C)CNC(C1CC(C)(NC(C2CCCS2)=O)C1)=O C(CNC(C)=O)(CC=C)NC(COCCOCC#C)=O.C(c1ccco1)=C(C(=O)N)C C1(NC(C(C)O)=O)(CNC(c2ccc(CSC(F)F)o2)=O)CCC(C)(C)CC1 c1(COCC)nc(C(=O)NC2(C)CC(NC(=O)C(C)c3ccsc3)C2)cs1 N1CC(C)CN(C(=O)C2=NOCC2)CC1C.Cc1nc(Cc2ccco2)sc1C=O C(=O)(C1=CCCSC1)N1CC(CCC=C)(C(N2CCC(CCCC)C2)=O)C1 N1(C(CC=CCC)=O)CC2CC3CC2C1C3NC(c1cc2c(cc1Cl)NCC2)=O Cc1cc(=NC(=O)C2CC23CCN(C(C2(C)CC2)=O)C3)[nH]n1C n1(CC(=O)NC2CC(N(C)C(C3CC3c3ccn(C)n3)=O)C2)cncc1C(=O)O C1(C(N2CC(NCc3cccc(C(=O)CBr)c3)C2)=O)COc2ccccc2O1 c1(C(N2CCCC(Cn3cc(C4CCN(C)C4)nn3)C2)=O)cnc(Cl)c(Cl)c1 C(=O)(C(C)(CC)OC)NCc1c(C(N(CC=C)CCC)=O)cco1 C1(C)(C(N2CC(NC(C=Cc3cccc(C)c3)=O)C2)=O)CC2(C1)CC(F)(F)C2 C1(C(=O)NC(CN(C(CC2N(C(C)=O)CCC2)=O)C)(C)C)CCC(=C(F)F)CC1 N1(C(C=Cc2c(OC)cccc2)=O)CC(NC(=O)C(F)(F)C(C)O)CC12CCC2 CC1(C)CC(CNC(c2ccoc2Cl)=O)CN(C(c2cnc[nH]2)=O)C1 C12(Nc3c(Oc4ncccn4)cccc3)CNCC(C3CCC3)(C1)C2 c1(C(N2CCC(F)(CNC(C=CSC)=O)C2)=O)ccc2nc(C3CC3)oc2c1 CC(C)CC(C(=O)N(CCC(=O)NOCCOCCF)C(C)C)C(C)C c1(C(=O)NCC2CC(F)(CNC(C(C=C)(C)O)=O)C2)cc(O)nc(OC)n1 C1(OC)CC(O)CN(C(=O)CC2C3CCC(C3)N2C(C2CNC(=O)N2)=O)C1 N1(C(C2CCC(C)CN2C(C2COCCO2)=O)=O)CC(O)C(O)C1(C)C C1(NC(C=C(COC)C)=O)COC2(C1)CN(C(=O)Cc1cccc3c1OCO3)C2 C1(C(=O)NCCCCC(N)=O)CC2CCC2C1.CC1(C)C2C1CNC2=O c1(CNc2cc(C(=O)NC(C)C#N)n(C)c2)c2c(nn1C)CCC2 N1(C(C2C(CC)CCO2)=O)CCN(C(=O)Cc2c(C)cnn2C)C2(CC2)C1 c1(CC)[nH]nc(C(=O)N(CC(C)(C)NC(C2C=CCS2)=O)C)c1C C12(NC(C=CC(CC)=CC)=O)CC(NC(=O)CC3CCCN3C(C)C)(C1)C2 C(=O)(C1=CCSC1)N1CC(OCCNC(=O)COCC(F)F)C1 c1(OCC)nc(=NCC(C(C)(C)C)NC(=O)C(C)C(C)(C)C)[nH]cc1C CCCCC(O)CC(=O)N1CCN(Cc2cc(C3(C(=O)NC)CC3)c(C)o2)CC1 c1(C(N2CC3(CC(NC(C4(SC)CCC4)=O)C3)C2)=O)ccc2c(O)ncnc2c1 CC1CN(C(=O)C(C)(C)N(C)C)CC1(C)CNC(c1ncncc1Cl)=O c1(C(N2CCC(NC(CC(=O)NCC#C)=O)CC2C)=O)c(OC)ncc(Cl)c1C c1(C(N2CC(COC)(NC(=O)Cc3c[nH]nc3O)C2)=O)cc(C(C)C)nn1C C12(CNC(CNS(CCOCC)(=O)=O)=O)CCC(CN(C(=O)C(C)N(C)C)C1)C2 C1(CC(=O)NC2(C(=O)OCC)CCCCC2)CCCCN(C(=O)CSC)C1 Cc1ccc(F)c(C(N2CCCC(CO)(NC(C3CCS3(=O)=O)=O)C2)=O)c1 C1(CCC(=O)NCC(F)CO)CCCN1C(c1c[nH]nc1Cl)=O c1(CC(=O)NCCC2CCCN(C(C(C)OCC(C)C)=O)C2)c(Cl)cccc1Cl N1(C(C=CCC)=O)CC(NC(c2ncc(F)cc2N)=O)CC12CCOC2 C(CCC(=O)NC1CC(F)(Cc2cn(CO)nn2)C1)NC(=O)OC(C)(C)C N1(C(CCC=C)=O)C2CCC1(c1cn(-c3ccc(COC)cc3)nn1)CC2 CC1CCc2ncc(C(=O)NC3(CCNC(C4CC4[N+](=O)[O-])=O)CCC3)n2C1 C1(C(c2cn(C3CCCNC3=O)nn2)=O)CCN(CCNC(C(C)CF)=O)CC1 C(C1c2ccsc2CCN1C(=O)OC(C)(C)C)NCc1n(CC)nc(C)c1 N1(C(c2cc(CC)nn2C)=O)CCC12CCN(Cc1ccc(F)cc1O)CC2 N1(C(c2c(C)ncn2O)=O)C2CCC1CC(NC(C1CN(C)CCO1)=O)C2 N1(CCN(C(C(CC(C)C)ONC=O)=O)c2cc(C)on2)CCC(O)C(C)(O)C1.CO c1(C(=O)NC2C3(CC(NC(C4C(C)C4)=O)C3)C2)cc(S(N)(=O)=O)c[nH]1 N1(C(C2(NC(C)=O)CCC2)=O)CCN(CC(N2CCC2C(C)C)=O)CC1 CCC(C(=O)NCc1ccc(CNC(C2CCCS2(=O)=O)=O)cc1F)C(C)(F)F C(C)(C(=O)N(C(C)CNC(C1CCCS1)=O)C)SCCCC N1(C(c2c(C)nco2)=O)CC2CCC2(CC(=O)N(CCC(F)(F)F)C)C1 c1(C(=O)NCC(CC)NC(c2cc(CO)n(C)n2)=O)cc(F)cc(Br)c1 C1(CNC(C2NC(=O)OCC2)=O)CN(C(c2ccc(CO)o2)=O)CC12CCC2 Cc1ccc(C(N2CC(NC(C3CC4(C)CC3CO4)=O)C(C)(C)C2)=O)c(C)n1 C1(C2(O)CN(C(=O)N(C)CCO)C2)(CNC(c2cc(COC)on2)=O)CC1 C1(C(N2CCC(OCCNC(=O)C(F)C3CCC3)C2)=O)C=CC=CC=C1 N1(CCCNc2nn(CC)c(C)c2)CC(C)CC(C)C1 C(=O)(CC1=CCCC1)NCC1(F)CCC(NC(C(C)Cc2cccnc2)=O)C1 c1(C(=O)NC(C)C(C)(C)NC(c2cnc(N(C)C)s2)=O)nn(C)c(Cl)c1Cl c1(CC(C)CN2CCN(CC(C)O)CC2)cccc(Cl)c1 CC1C(NC(C2(C)CCSCC2)=O)CCN1C(c1cccc(OCC(N)=O)c1)=O C12(C(=O)NCC(CCCC)O)CCCC1CCN2C(C1CC2CCCC2C1)=O c1(OC)cc(C(=O)NC(CC2CCC2)C(=O)NCc2nc(C3CC3)n[nH]2)[nH]n1 N1(C(CCCC#N)=O)CCC(c2cccs2)(CNC(C2CC23CC(O)C3)=O)CC1 Cc1ccc(S(=O)(=O)CC(=O)NCC2CN(C(c3cscc3C)=O)C2)cc1 CCC(CC)(C(=O)N1CCCC1Cn1cc(CNC(=O)C(C)S(N)(=O)=O)nn1)C(C)C CC(C)CC(C)C(=O)N1CCC(CC(N2CC(O)C(O)C2)=O)C1(C)C C1(C(N2CCCC(CCNC(=O)CCC3CCCO3)C2)=O)CCc2nncn2C1 C1(C(=O)NC(c2n(CC)ccn2)C)CN(C(=O)CSC2CC2)CC(C)O1 Cc1cc(C)c(C(N2CCCC(CNC(=O)C(C)Cn3cccn3)C2)=O)c(=O)o1 C1(NCCONC(CC2(NC(c3cc(OC)n(C)n3)=O)CC2)=O)COCC(=O)N1C N1(C(CCC(=C)Cl)=O)C2CCC(C2)C1C(=O)NCC(C)CO c1(C(N(CC#CC)C)=O)cn(CNC(C2(CCF)CCC2)=O)cn1 C=C1CCN(C(=O)C(CSC)OC)C(C(=O)NCC2CC3CCC(C2)C3)C1 N1(C(=O)Cc2c[nH]nc2O)CC(NC(C2COCC2C(F)(F)F)=O)C2(CC2)C1 C1(N(C(CC=CC)=O)CCF)CCCN(C(c2cc(N3CCCC3)ncn2)=O)C1 N1(C(CCNC(Cc2ccc(C)nc2)=O)=O)CCN(C)CC1C1CC1 C(CCC(C)(C)NC(=O)CCNC(C1CCC1)=O)NC(C(N1CCC(C)C1)=O)=O N1(C(C2C(C)(Br)C2)=O)CC2(CCN(C(c3ccc(C4CCOC4)cc3)=O)CC2)C1 N1(C(C2N(CCCC)CCOC2)=O)CC2(CCN2C(=O)CCC2CCCO2)C1 C1(CNC(CC(C=C)C)=O)C2CCC(C2)N1C(c1cccc(C2(C)CC2)c1)=O c1(CC(=O)OC)ccc(S(=O)(=O)NC2CC3CCC(C2)N3C)cc1 CCC(C)C(CN=c1[nH]c(=NC2CCS(=O)(=O)CC2)[nH]c2cc[nH]c12)OC C1(C(N2CC(C(=O)NC3CCCC3)(COC)C2)=O)CC12CCOC2 c1(NCc2c(Br)c(C)n(C)n2)ccc2ccc(Cl)c(Cl)c2n1 S(=O)(=O)(c1ccccc1)NC(C(=O)NC1CCN(C(COC)=O)C12CC2)C c1(C(=O)NC23CC(CNC(C4(CC#C)CCCC4)=O)(C2)C3)cnc2ccnn2c1 CC(O)C(F)(F)C(=O)NCCCN(C(=O)Cc1cc(Cl)cs1)CC1CCCC1 Cc1cc(-c2cn(C3CC(C(=O)Nc4cc(Br)ccc4C)C3)nn2)c(F)cc1Cl CCC(CC)CC(C(=O)Nc1cccc2ccccc12)N(CCC#N)CCSC c1(C(=O)NC(C(=O)N(C(C=C)C2CC2)C)C2CCOC2)sncc1C CC(C)CC(CN(C)C)NC(=O)CNC(=O)C(C)(CC)ON C(C)(CNC(c1c(F)cccc1F)=O)(CC(C)C)NC(COC(CC)C)=O C1(CC)CC(C)(C)CCN1C(C1CC(n2cc(CCC(=O)O)nn2)C1)=O c1(OCC)cccc(C)c1NC(C1CC(NC(=O)CCc2ccncn2)C1)=O N1(C(CC)CC)CC(C(N2CCCCC2CN(C(=O)CC(C)C)C)=O)CC1=O N1(C(CSCC#C)=O)CCN(C(=O)CCCc2ccc(C(C)C)cc2)C(C)C1C N1(C(C23CC(C(=O)O)(C2)C3)=O)CCCC(CC(=O)NC2(CC#C)CC2)C1 CCC(N=c1[nH]c(Cl)nc2cc(C)sc12)C(OC)CNC(=O)OC(C)(C)C c1(OC)cccc(CO)c1-c1cnc(C(=O)N(CCO)CCO)cc1C S(=O)(=O)(c1ccc(C#N)c(NC2CC(C(F)(F)F)C2)c1)N1C(C(C)O)CCCC1 c1(C(N2C(C)CC(NC(C3(COC)CC=CC3)=O)C2)=O)cnc2ccnn2c1O C1(NC(C(C)OCCC#C)=O)CCCCN(C(c2ccc(C#N)[nH]2)=O)CC1 c1(N2CC(NC(=O)CSc3ccccn3)CC(C)(C)C2)ncnc2[nH]c(Cl)cc12 Cc1ncc(C(N2CCC(CN(C(c3ccsc3Cl)=O)C3CC3)CC2)=O)n1C c1(C(=O)NC(CNC(C2CCC3(CCC3)CO2)=O)CO)nnn2c1C(=O)NCC2 C1(NC(c2cnco2)=O)CCN(C(C2CC2c2cccc(Br)c2)=O)CC1 CC1(C)CN(C(C2(C)CCCO2)=O)CC1CNC(c1ccnc(CO)c1)=O Cc1ccc(C=CCC(=O)NC2(CCCNC(=O)C(C)O)CC2)cc1 O=S(=O)(c1ccc(NC2CCCOC2CC2CC2)c(Br)c1)N1CCC2(CC1)CC2 C#Cc1c[nH]nc1C(N1C(CNC(=O)CCc2cncc(OC)c2)CC2CC12)=O C(=O)(C1CCc2c[nH]nc21)NCCc1c(C(=O)NC2(C)CC(N(C)C)C2)c[nH]n1 C1(NC(CN(C(C)=O)C)=O)CN(C(C2COC(C)(C)C2)=O)CC2(CC2)C1 C1(NC(C(CCC)NC(=O)CCCN(C)C(C)C)=O)CCCCC12CC2 C(CC(F)(F)CO)NC(CN(C)C(c1cnn(C)c1Cl)=O)=O N1(C(CN2CCCC(NC(C)=O)C2)=O)CCN(C(C23CC(C2)C(C)O3)=O)CC1C C1(C(=O)NC2(CN(C)C(C3CC(n4cnnc4)C3)=O)CC2)CCC(C)(O)CC1 c1(C(=O)NC2CCN(C(=O)CC3OCCCO3)CC2O)cncc2nc(O)[nH]c12 C1(NC(c2n(CC)ncn2)=O)CCC2CC1CN2C(c1ccccc1C)=O C1(CC(N2CCCC(N(C(C(C(C)C)O)=O)C)C2)=O)CCC2(CC1)OCCO2 c1(CC)cc(C(=O)NC2CCCC2NC(=O)CC2CCCCO2)ccc1O Cc1cc(F)c(CN2CCOCC2C(=O)NCC2CCC(F)(F)C2)c(Br)c1 Cc1cccc(CC(N2CC(NC(=O)C=CC3CCCC3)C(C(F)F)C2)=O)c1 c1(CN2C(C(N(C)CC3CCCN3C)=O)CC2)c(I)ccnc1F N1(C2CCCN(C(CCNS(C)(=O)=O)=O)C2)CCN(C(C2(O)COC2)=O)CC1=O c1(C(=O)NCCC2(O)CN(C(C(CN(C)C)O)=O)C2)ccc(O)cc1C(F)F C12(C(=O)NC3CCC(C)CC3)CC(CN(C(=O)CCC3CCCOC3)C1)C2 c1(C(N2C(CNC(C3CC4CCC4C3)=O)C=CC2)=O)ncc(Cl)cc1Cl c1(C(=O)NCCCN(C(=O)C(O)C2CCC2)C)ccc(Cl)c(O)c1N C1(NC(CN(CCCN(C)C)C)=O)CC(NC(=O)CCC(C)(C)F)C12CCC2 Cc1[nH]nc(C(=O)NC2(CO)CN(C(C3C4CN(CC(F)(F)F)CC34)=O)C2)c1O c1(C(N(c2cccc(C#N)c2)CC)=O)ccc(Br)cc1C#N C(=O)(C1CC(=O)Nc2ccccc21)N1CCN(C(CCOCC)=O)CC1CCO Cc1cnc(-c2cn(CC3CCCN3C(=O)C(F)CN(C)C)nn2)c(C)c1 N1(C(c2cc(C)oc2C)=O)CCCC2CN(Cc3cccc(C#N)c3)CCC12 C1(C(N(C(CC)CC)C)=O)COCCN(CCC(=O)NC2CC2)C1 N1(C(c2c(COC)cco2)=O)CCC(c2nc(-c3cc(Cl)ccc3F)no2)CC1C C(C(C)(C)C(F)(F)F)Cc1n(CC=C)nc(-c2ccc(OC)nc2)n1 C1(NC(C(C)OCCOC)=O)C2COCC1CN(C(=O)CCCC#N)C2 c1(CCOCC)nc(C2CCOC2)nn1C12CC(C3CCCCC3)(C1)C2 C1(C(N(CCC(=O)NC2CC(C(N)=O)C2)CC#C)=O)CCN(C)C1C c1(CC(=O)N(C2CN(C(COCC=C)=O)CC2(C)C)C)c[nH]c2c(F)cccc12 C1(CNC(C(CC)N(C)C)=O)CC2COCC2N1C(C1CCC(N(C)C)CC1)=O CCC(C)C(O)CC(=O)NCC1(NC(=O)C(=O)NC2CC2)CC(F)(F)C1 C#Cc1cccc(CC(=O)NCCNC(c2ccc(C(=O)C3CC3)cc2)=O)c1 N1(C(C(=Cc2ccncc2)C)=O)CCOC2(CCN(C(=O)C3=CC(C)(C)C3)C2)C1 C(=O)(C(CCSC)NC(C1(CC2CC2)CC1)=O)N(C)Cc1n(CC)ccn1 N1(C(Cc2ccc(NC(C)=O)cc2)=O)CCC2CN(C(=O)CCCCBr)CCC12 N1(C(C(N2C(CC)CCC2)=O)=O)CC2(CCN(C(C3CN(S(C)(=O)=O)C3)=O)C2)C1 C(=O)(CCC(C)NC(=O)Cc1ccsc1)N(C(C(=O)OCC)C)C N1(C(C(C2CC2)OC)=O)CC2(CC(NC(C3(C)CCC3(C)C(=O)OC)=O)C2)C1 c1(C(=O)NC(c2ccccc2F)C)c(-c2cnn(C(C)(C)CO)c2)cncc1F N1(C(CC2(NC(C(C)NC(C)=O)=O)CCC2)=O)CCCC(F)(F)C1 C(=O)(C1=Cc2ccccc2C1O)N1CCC(C=C)(C(=O)OC(C)(C)C)CC1 C(=O)(C1CCc2nccn21)NC1C(C(=O)NCc2c(C)cc(F)cc2)OCC1 CCC(F)(F)C(C)(C)NC(C1CN(C(c2ccc(SC)o2)=O)CC12CC2)=O c1(C(=O)NCC(C)NC(c2ncoc2C2CCC2)=O)cnc(O)c(Br)c1 c1(C(N2CC(CCCNC(C(C)SC)=O)OCC2)=O)c(O)cccc1F c1(NC(C23C(NC(C(C)C4CCC4)=O)C4CC2C3C4)=O)cccc2ccccc12 C1(N)CC2(C1)CC(N)C2.C(=O)(C(F)CC1CC1)C(c1coc(C2CCC2)n1)=O CC1(C(=O)NC2CC(F)(CNC(=O)C(O)Cc3cnc[nH]3)C2)CCOCC1 c1(C(C)NC(=O)C(C)(F)C(=O)O)ccc(F)cc1F N1(C(CC2(CNC(c3coc(C(F)F)c3)=O)CC2)=O)CCC(O)(CO)C1 c1(C(=O)NCC(C)(C2CC2)NC(=O)Cn2nnc(=O)[nH]2)ccccc1[N+](=O)[O-] Cc1ccc(C(=O)NC(C)CCN(C)C(C2C=CCS2)=O)s1 C(=O)(CS(=O)(=O)CCC(F)(F)F)NC1CCC(CCNC(c2c(C)ccs2)=O)C1 C1(C#N)(C(=O)NC2CCN(C(C3(C)CC(C)(C)C3)=O)C2)CCCCC1 N1(C(C(Cc2cnc[nH]2)OC)=O)CC2(CC2)CC1C(=O)NCCC1CCN(C)C1 c1(C(=O)NC(CCNC(C2(CCC=C)CCCC2)=O)C)ccc2ocnc2n1 N1(C(c2ncnc(C)c2C)=O)CC=C(CC(=O)N(C)Cc2cn(C)nn2)CC1 Cc1cnn(C)c1CC(=O)NC(C)CCCNC(C1CC1C(F)(F)F)=O c1(C(=O)NC(C(C)NC(=O)CCn2ccnc2)(C)C)cc(=O)n(C)cn1 C=CCC(CC(F)F)C(=O)NC1CN(C(C2(Cl)CC2)=O)CC1O c1(C(C(=O)NC2(CNC(C(F)=CCC)=O)CC2)=O)c[nH]c2cc(F)ccc12 N1(C(C)C)CCCC1C(=O)NC12CC(NC(=O)Cc3csc(S)n3)(C1)C2 c1(C(N2CCC(CNC(C3C(C)(C)CO3)=O)CC2)=O)cc2cnccc2[nH]1 CC(c1ccsc1)=CC(=O)NCC1CC(NC(C2(C#N)CCOC2)=O)C1 N1(C(c2csc(C)c2N)=O)CCCC(N(C(=O)C2=CCCCC2)Cc2ccccc2)CC1 N1(C(C(C)OC2CCCC2)=O)CCC2(COC(CNC(C3(O)CCC3)=O)C2)C1 CC1(C2CC2)CN(C(=O)C=CCNC(C2(N(C)C)CCCCC2)=O)CCO1 c1(C(=O)NCC(CCNC(C2CC(C)=C(C)CC2)=O)O)cc(F)cc([N+](=O)[O-])c1 c1(C(=O)OC)cc(C(N2CCCC(NC(=O)CN3CC4CC4C3)C2C)=O)ccc1O C(=O)(C1=CCCCC1)N1CC=C(CNC(C2(C(=O)OC(C)(C)C)CC2)=O)C1 CN1CCCC(C(=O)NCC2CCCN(C(c3cc(-n4ccnc4)cs3)=O)C2)C1 N1(C(C=COCC)=O)CCN(C(c2cnc(N3CCOCC3)s2)=O)CC(CO)C1 Cc1nn(C)cc1C(=O)NC1CC(F)(CNC(c2ccnn2C)=O)C1 C(C(CNC(C1NC(=O)OC1(C)C)=O)S(C)(=O)=O)NC(c1n(C)cnc1)=O C#Cc1cccc(C(=O)NC2CC3(C2)CC(CNC(=O)COC2CCC2)C3)c1 CC1CC(C(=O)NC2CCN(CCF)C2)CN(C(=O)C=Cc2nccs2)C1 C(C(O)CNC(c1cccs1)=O)N(C(=O)COCCF)C Cc1cc(C)oc1CNC(=O)CO.c1(CN(CCOC)C(C)C)cccnc1 C=Cc1cncc(C(=O)N(C(C)C(N2CC3(CSC3)C2)=O)C)c1 N1(C(COCCCC)=O)CC2(CC(NC(C3CCC(O)CN3C)=O)CO2)C1 C12(CNC(C(C)CF)=O)CCCCC1N(C(c1ccc(CC#N)cc1)=O)CCC2 c1(C(=O)NC(C2N(C(CC(CC)C3CCC3)=O)CCC2)C)cnc(O)c(F)c1 Cc1cc2[nH]c(C(=O)NC3COCC3NC(C3CC(=O)N(C)C3)=O)cc2s1 C12(CNC(=O)CC3CCCO3)CCCOC1CCN(C(=O)Cc1cn[nH]c1)C2 c1(C(=O)OC)ccc(C(C)NC(C(F)(F)F)c2cccnc2)nc1 C1(OC)CN(C(=O)CC(c2cccc(F)c2)C)CC1NC(=O)Cc1nccn1C Cc1c(CN2CCCCC2c2ccc(Br)cc2)cnn1C(C)C C(=O)(CC(C)(C)NC(c1cc(OC)ns1)=O)NC(C#C)C C1(C(=O)NCC2(C)CC(O)C2)CN(C(=O)CCC2CC2)CC12CC2 C1(CO)CN(C(=O)CCc2cnccn2)CC1C(=O)NCC1(CCO)CCCC1 CCC(C(=O)N(C)CCOCCNC(=O)C=CC(C)=O)C(C)(C)CC c1(OC(C(=O)NCC(C)NC(c2cc[nH]n2)=O)(C)C)ccc(CO)cc1 CC1(CNC(=O)CC2(C(F)(F)F)SCCS2)CCCN1C(C1CCCSC1)=O C1(N(C(=O)CC2(O)CCC2)C)CN(C(C2(C)CC(F)(F)C2)=O)CC1O c1(SC)cn(C)nc1CNC(=O)CC1CCN(C(c2ncccc2F)=O)CC1 CC1(NC(=O)CCSCC(N)=O)CN(C(=O)CC2C=CCC2)C1 c1(C(=O)NC(CN(C(C(F)=CCC)=O)CC)C)cc2c(C)cc(C)cc2[nH]1 Cc1nc(N(C)CC2CCCCN2C(C2CCCCC2O)=O)c(Cl)cc1C#N Cc1nn(C)c2cc(NC(C3CC34CCN(C(=O)Cn3ccnn3)C4)=O)ccc12 c1(CC)cc(C(=O)NC2C=CC(CNC(=O)C(C3CCC3)OC)C2)n(C)n1 c1(C(=O)NCCCC(C)NC(C2(C#C)CCC2)=O)c(C)ccnc1C N1(C(c2cccc(-c3cncnc3)c2)C(=O)NCC2CC2)CCN2CCC1C2 CC1(NC(=O)CNS(=O)(=O)C2CC2)CN(C(c2ccc(C(F)(F)F)s2)=O)C1 N1(C(c2c(C(C)NC(c3cc(=O)cc[nH]3)=O)noc2)=O)CCC(F)(F)C(O)C1 c1(C(=O)NC2CCC(CCNC(CC3NC(=O)OC3)=O)C2)ncncc1Cl C1(NC(C=CC(C)C)=O)CCCC1NC(=O)C(O)Cc1cn(C)cn1 CC1C(NC(=O)CCCN=[N+]=[N-])CCCN1C(C1COC(=O)C1)=O c1(C(=O)NC2CCC(CCNC(COC)=O)C2)nn2c(c1C)CCCC2 c1(C(=O)NC(CNC(C(CCC)N(C)C)=O)C)ccn2[nH]c(=N)nc2c1 C(=O)(CC(c1ccccc1)N(C)C)NCC(C)N(C)C(c1csc(CO)n1)=O N1(C(c2ccc(C)c(Cl)c2F)=O)CC(CO)C2(C1)CN(C(=O)CC(C)C(C)C)C2 N1(C(C2(C)CCCN2C(=O)CCOCC(F)F)=O)CCCC2C(=O)NCC12 c1(C(N2CC(NC(C=CCCC)=O)C(C)(C)CC2)=O)ccc2cccc(Cl)c2n1 c1(CC)nocc1C(=O)NCCc1ocnc1CNC(C1CC1CC(C)C)=O C1(CNC(CCC=C)=O)CCC(C)(C)CN1C(=O)CCN(CC(C)C(C)C)C Cc1cc(C(=O)NCC2(NC(=O)C(c3ccc(Cl)cc3)CO)CC2)ncc1Cl C(CC(C(=O)NCC1CC1NC(=O)CSCc1cccc(C(N)=O)c1)OC)OC N1(C(C(c2ccc(C)o2)C)=O)CC(O)C(O)C1CNC(c1occc1C)=O c1(NC2CCC(C)(C)CC2)ccc(S(=O)(=O)NCC2(CCO)CCOC2)cc1F Cc1cncc(C=CC(=O)NCCC2CCN(C(=O)C(C3CCCCC3)F)C2)c1 C12(C(=O)NC(C(=O)NCC3(CC)CCC3)C)CCC(CC1)CO2 C1(NC(c2cccc(OC)n2)=O)CN(C(=O)CC2COC(=O)N2)C2(CCC2)C1 c1(C(c2nnnn2CCC2(C)CC2)NCC(C)CO)ccc(Cl)c(F)c1F N1(C(CCC=C(C)C)=O)CCC2C(CCCN2C(c2sc(C)cc2C)=O)C1 C(=O)(C(CCCOC)NC(=O)C(C)N=[N+]=[N-])NCCc1cc(CC)no1 N1(C(CC2CCC(C)(C)O2)=O)CCC2CC1CN(C(=O)CC1=CCCCC1)C2 c1(C(=O)OC)ccc(S(=O)(=O)Nc2ccc(OC)nc2OC)n1C CN1CCN(C(C2CCCSS2)=O)CC1CNC(=O)CC1CC2CC2C1 Cc1nc(C(F)(F)F)oc1C(=O)NC1CC(CNC(=O)CC(C)c2ccco2)C1 C1(C(=O)NC(C2CCN(C(C3CC(=O)N3)=O)C2)C)C2CCCCCCC12 c1(C(=O)NC(C2CN(C(=O)CN3CCCC3=O)C2)C)cnc2ccccc2c1 N1(C(c2cccc(OC)c2)=O)CCC2(CCCN(C(c3cnoc3C)=O)C2)C1 C(C(C)(C)C(C)(C)O)NC(C(CNC(c1coc(C(N)=O)c1)=O)OC)=O c1(C(=O)NCC(C)NC(c2c(F)ccc(C)c2O)=O)cccc2c1OCC2C c1(NCCCc2c(C)cccn2)ccc(S(=O)(=O)N2CC3CC=CC2C3)cc1Br C1(C)(CNc2cc(C)oc(=O)c2)CC(C2CC2)=NO1 Cc1ccc2oc(C(N3CCC4(CC3)CCN4C(C3CC3C3CC3)=O)=O)cc2n1 C(=O)(C1CCc2c[nH]nc21)NCC(CNC(=O)CC(C)(C)C(F)(F)F)OC CON(CCO)C(=O)C1CC(NC(=O)CC2CC(C)C2)C12CCC2 c1(C(N2CC3N(C(CC(C=C)C)=O)CC(C3)C2)=O)c(C)c(C)nn(C)c1=O N1(C(COCC=C)=O)CCc2ccccc2C1CNC(=O)CSCCN(C)C c1(CC(=O)NCC2(C)CC(NC(=O)C3=CCCOCC3)C2)ccccc1[N+](=O)[O-] C1(C(N2CC(F)(CNC(C3(CN(C)C)CC3)=O)C2)=O)CC12CCSCC2 N1(C(C)=O)CSCC1C(N1CCC(C(C)N(C(=O)C(c2cccnc2)C)CC)C1)=O C1(C2(O)CCN(C(C3(C)CC3(F)Cl)=O)CC2)(NC(Cn2c(C)nc(C)n2)=O)CC1 N1(C(CSCC#C)=O)CCC23CN(C2)C(=O)C13.N1(NC(=O)OCC)CCOCC1 C1(C(=O)NCC2C(CNC(C(CC)N3CCCC3=O)=O)C2)CC2CCC(C1)O2 Cc1coc(C(=O)NC(C2CCN(C(c3cncc(C(N)=O)c3)=O)C2)(C)C)c1C c1(SC)ccc(CC(N2CCN(CC(C)NC(=O)CC3CCCO3)CC2)=O)cc1 C(=O)(N=c1ccnc(C(F)(F)F)[nH]1)C1N(C(C2CC=C(C)CC2)=O)CC(F)(F)C1 C1(C(N2CCCC2CN(C)C(C2(C)CNC(=O)C2)=O)=O)(OC)CCCCCCC1 C1(C(=O)NC(C(C)C)CNC(c2c(C(F)F)cnn2C)=O)Cc2ccccc2N1 N1(C(c2c(OCC)nccc2)=O)CCOCC(C)(CNC(C2C(C)C2(F)F)=O)C1 CC1C(NC(=O)CC(=O)NC2CC2)CC2CCC1N2C(=O)CCN1CCCC1=O C1(CN(C(=O)CCc2cc(C)nn2C)CC)CCN(C(C2CN(C)C2)=O)CC1 C(=O)(C1COc2ccc(Cl)cc21)N(C)CC1(O)CCN(C(CCNC(C)=O)=O)C1 c1(C(=O)NCCC2CC(NC(CSC(C)C)=O)C2)ccc2c(c1)CCCS2 N1(C(c2cc(C)c(C)s2)=O)CC(C)(C)CC1CNC(c1cc(C(F)F)cs1)=O c1(CNC(=O)NCCC(O)CCO)cc(O)cc(O)n1 C1(C(=O)NCC(CNC(=O)C(F)(F)c2ccnn2C)OC)CCC2CC12 C1(C(=O)NCCC(C)NC(=O)CSc2ccccc2)CCC(C(=O)C2CC2)O1 C12CCCN(C1)C(=O)NS(=O)(=O)N2.N#CCCSC(C)(C)C C1(NC(=O)NC(C23CCC(CC2)C3)C)CC12CCCCCC2 Cc1cc(C(N2CC=C(CNC(c3cc(Cl)cnc3O)=O)CC2)=O)cn(C)c1=O N1(C(CCC=C)=O)CC(CNC(=O)Cc2ccc(Cl)cc2)OC(C)(C)C1 c1(C(N2CCC(N(C)C(C3CC3C(F)(F)F)=O)C2)=O)cnc2cc(O)ccc2c1 n1(CCOC)nc(-c2cncc(Br)c2)nc1C1CN(C)CC1C O=S(=O)(c1cccnc1N1CCC(O)C(F)C1)NCc1cn(C2CC2)cn1 N1(C(CC(CC)SC)=O)CC2CCCC2(C(=O)NCc2ccc(O)cc2F)C1 Cc1ccc(C(N2CC(NC(C3(C)CC(C)(C)C3)=O)C(O)C2)=O)nc1 CC1(C(=O)NCCC2CCC(NC(C3(Cl)CC3)=O)C2)CC2CCC(C1)S2 C1(O)(C(=O)NC(CN(C(C)C)CC)C)CCCN(C(=O)C(=O)NCC(F)F)C1 CN1CC(NC(C2CCC(NC(=O)Cc3ccc(O)cn3)C2)=O)C(C)(C)C1 C(CCC(=O)N(C(C)CCNC(=O)C(c1ccccn1)C)C)=CCC=C C12(C(N3C(C)CSCC3)=O)COCC1CN(C(=O)CCN1CCCCC1)C2 c1(CC(=O)N(C2CCC(NC(CC=CC=C)=O)C2)C)c[nH]c2c(Br)cccc12 C1(NC(CCC2CCC(C)O2)=O)CC2(C1)CC1(CC(NC(=O)C=CCO)C1)C2 c1(C(=O)NCC2CC(NC(c3ncc(SC)s3)=O)C2)ccc(OCC(F)F)nc1 N1(C(C(CNC(C(C)(C)OC)=O)N(C)C)=O)CCc2ccsc2C1 Cc1ccccc1C1CN(Cc2ccns2)CCN1 N1(C(CC2CC(=C)C2)=O)CC2C(N(C(=O)C(=O)NCC(F)(F)F)C)C2C1 C1(NC(CC(C=C)C)=O)CCC2(CCN(C(=O)C=CC(=O)NC3CC3)CC2)C1 n1(CC#C)c(C)cc(C(=O)N(CCC)CCNC(=O)C(C(C)O)NC(C)=O)c1C N1(C(C(C)(N(C(CCCOCC)=O)C)C2CC2)=O)CCC(CO)C(C)C1 C(CC(=O)N1CC(CS(C)=O)C1)(CC(C)C)NC(CCCCNC(C)=O)=O CC(C)C(O)C(F)(F)C(=O)N1CCCC(N(CCF)C(c2cccn2C)=O)C1 c1(C(=O)NC2CN(C(Cc3nc(C)[nH]n3)=O)C(C)C2)nc(O)nc(O)c1F Cc1cc(C(=O)NC2CN(Cc3c(O)cc(F)cc3F)CC2(F)F)cc(C)c1F c1(C(N2CC(NC(CCCCOC)=O)C(OC)C2)=O)cnc2ccccc2c1 c1(CC)onc(C(=O)NCC23CC(NC(c4cnc(C5CC5)[nH]4)=O)(C2)C3)c1C C(N=c1[nH]cnc(Cl)c1Br)C1OCC(CNC(c2c(CCC)n[nH]c2)=O)C1 CC1CC(C)CN(CCN(c2ccccc2C(=O)OC(C)(C)C)CCO)C1 S(=O)(=O)(c1ccc(C(N)=O)cn1)NC(CCC)C1CCCC1 C#CCC(C(=O)C(=O)C=Cc1cn(C)nn1)NC(=O)CCC1CC(N(C)C)C1 C12(CNC(C=NOC)=O)CCC(CC1)N2C(=O)CC1CCCC(C)(C)C1 c1(C(=O)NC2C(NC(c3cccc(C)c3N)=O)CC2)ncccc1S(C)(=O)=O CCC1CN(C)CC2CCN(C1=O)CC2.C(=O)CC(C)OC.OC N1(C(C(CCC)CNC(=O)C=CC2CCCN2C)=O)CC2(CCN(C)CC2)C1 C1(CNC(C(C)OCC)=O)CCN(C(C2CCN(CC(C)C)CC2)=O)C12CCC2 C#CCC(C)(C(=O)NC12CCC(C1)OC2C)NC(C1CCC1OCC)=O c1(C(=O)NC(C(C)NC(CN(CCC)C)=O)C)c(OC)cc(OC)cc1CC C(=O)(CC(C)(C)C=C)NC(C(=O)NCC=C=C)Cn1cccn1 CC1(C(=O)NCCOCCNC(c2ccc(CN(C)C)o2)=O)CC2CCC1O2 N1(C(c2cc(CC)[nH]n2)=O)CC2CCC1CC2NC(=O)CCc1cn(C)nc1C CCC(CC)CC(=O)N1CC(N(C(=O)Cc2csc(-c3nc[nH]n3)n2)C)C(F)C1 c1(CCCCNC(COC)CCc2ccccc2)ccc(Cl)cc1 Cc1cnc(C(=O)NCC(C)(C)CCNC(c2ccc(C(N)=O)cn2)=O)c(F)c1 c1(C(=O)NCC2C(NC(C3CC4(CC(=C)C4)C3)=O)C2)oc2c(c1C)C(=O)CCC2 CC(CC1CCC1)C(=O)NCC1CCN1C(c1nn[nH]c1Cl)=O N1(C(c2csc(C)c2C)=O)CCC2CN(C(=O)C(C)(C)CC3CC3)CCC2C1 C=CCC(CC(=O)NCC(O)CC(=O)OC)NC(C1(C)CC(C)=NO1)=O c1(OCC2CC(NC(C3(F)CC(NC)C3)=O)C2)ccc(Cl)cn1 N1(c2nnc(-c3c(C#N)cccc3)n2CC2CC2)CCn2ncc(Br)c2C1 c1(SC(CCC(=O)OC)Cc2ccccc2)ncnc2[nH]ccc12 C1(N2CCOCC2)(C(N(CCC(C)NC(C2C(CC)C2)=O)C)=O)CCCC1 N1(C(C2N=C(C)SC2)=O)CCC(C2(NC(=O)CC3=NNC(=O)C3)CC2)C1 Cc1cn2c(CCC(N3CC(O)(CNC(=O)Cc4ccccc4)C3)=O)csc2n1 C(=O)(C1COc2cc(C)c(C)cc21)N1C(CCNC(CCCOC)=O)CCC1 N1(C(C(C=C)CC)=O)CC(N=[N+]=[N-])CC1C(=O)NCC1(CO)CC1C=C N1(C(C(C2CN(C(C)=O)C2)O)=O)CC2C(C1)C2(F)F.C1CC1(C)C(F)F C1(C(N2CC(CCC)OCC2)=O)CNC(=O)CN1C(c1cc(C)sn1)=O CCCC(CCC)C(C)(c1nnnn1C(C)C)NCCCC=CC c1(NC(C(=O)NC2C(C#C)CCC2)=O)ccc(Br)nc1C(F)(F)F C(N=c1nc(C)c(Br)c[nH]1)C1(NC(c2c(C)coc2)=O)CCCCC1C c1coc(CNCCNCCC2CCSC2)c1 C(=O)(C(C)C(C)(F)F)N1C(CNC(C(=Cc2cccs2)C)=O)CCC1 N1(C(C(CN(C(c2c(CCC)nco2)=O)C)C)=O)CCCC12CCNC2=O c1(C(=O)NC2CC(CCNC(C3(N4CCCC4)CC3)=O)C2)cn(C2COC2)nn1 Cc1ccccc1CC(=O)N(C1CN(C(=O)C(C)C#N)CC1O)C N1(C(c2ccc(C(=O)OC)nc2)=O)C(C)C2CC1C2NC(c1cc(C)oc1C)=O Cn1nnc2cncc(C(=O)NCC=CCNC(c3cc4c(s3)CCOC4)=O)c12 c1(C(=O)NCC(=C)CCNC(c2cccc(Cl)c2C)=O)nn(C)cc1[N+](=O)[O-] n1(C(C)C)ccc(C(N2CC(OCc3ccccc3)CC2CNC)=O)cc1=O N1(C(C(C=C)O)=O)CCCC(C2CN(C(c3cscc3C(N)=O)=O)C2)C1 C1(NC(C(=C)F)=O)CCC2(C1)CN(C(c1ccc(O)c(C(F)(F)F)c1)=O)C2 c12ncccc1N2C(=O)CN1CCSC1.c1(C[Si](C)(C)C)ccccc1 C1(NC(C(n2ccc(C)n2)C)=O)C=CCN(C(=O)CSCC(N)=O)C1 C1(C(=O)NC(c2cncs2)C)CCCCCCN1C(C1COCCC1C)=O C(=O)(C(C)(C)C(F)F)NCC(CN(C(CC1(COC)CC1)=O)C)C N1(C(c2n(C)c(S)nc2)=O)CC(CNC(=O)CC(F)(F)F)C(C)(C)C1 C1(C(=O)NCC2(NC(Cc3nnc(C)s3)=O)CCOC2)CCN(C2CC2)CC1 CC1(O)CON(C(=O)C2COCC3(CCC3)O2)C1.C=O N1(C(CN(C(=O)OCC)C)=O)CC(CC(=O)NCCN2CC3CC3C2)CC1C CC1CCN(C(c2ncn(-c3ccccc3)n2)=O)CC1NC(C1CC(F)(F)C1)=O N1(C(C(c2ccc(F)cc2)C)=O)CC(NC(c2ccsc2Cl)=O)C(C)(C)C1 c1(C(N2CC3C(NC(C(CC)OC4CCCC4)=O)(C3)C2)=O)cc2cccnn2n1 Cc1c(C(=O)OCC2CCN3CCC2C3)[nH]c2c(C)cccc12 Cc1cccc(C(N2CC(NC(=O)C=CCOCC(F)(F)F)CCC2C)=O)c1F C1(C(C)NC(c2c[nH]c(C(N)=O)c2)=O)CN(C(C2CCCC2C(F)F)=O)CCO1 C1(NC(C(OC)OC)=O)CN(Cc2ccc(CO)cc2)CC1C#N C1(c2nnc(N3C(C=C)CCC3)n2CC)CN2CCCN1CC2 c1(CC)nc(O)c(C(=O)NC2CCCCC2CNC(=O)Cc2cnco2)cc1C CC1(C(=O)NCC=CCNC(=O)CCn2cccnc2=O)COCCO1 CC1CN(C(c2ccc(N)cc2Cl)=O)CCC1CNC(=O)C(C)(C)COC(C)C N(C(=NCCCCl)NCc1cscc1C(N)=O)CC1C(C)C1(F)F c1(C(=O)OCC)nn(C2CCOCC2)cc1NC(c1ccns1)=O c1(CC)ccc(C(=O)NC2(C)CC(NC(C3CC3(C)C)=O)C2)c(O)c1 c1(C(N2CC(NC(C(COC)OC)=O)C2)=O)cc2c(F)c(Cl)ccc2[nH]1 CC1(C)CC(CNC(=O)CCC2(C)CC2)N(C(=O)COC(C)(C)C)C1 CC(=O)CCCC(C)C(=O)NCC1CC(NC(C2CCC(C)(C)C2)=O)C1 CCCCC(C(=O)NCc1nc(CNC(=O)C(F)C(F)(F)F)cc(O)n1)C(C)C C=Cc1cnn(C)c1C(=O)NCCCN(C)C(C1CC12CC(O)C2)=O N1(C(Cc2cc(C)nn2C)=O)CCN(C(c2cc(C)n(C)n2)=O)CC(C)(F)C1 c1(C(=O)NCC23N(C(COCCC)=O)CCC2CC3)cc2nc(Cl)ccc2s1 N1(C(C(C)OCCCCCC)=O)CCN(C(C23CC(CCO2)C3)=O)C2(CCC2)C1 N1(C(C(C)OCC=C)=O)CCCC1C1CCN(C(=O)CNc2ncccn2)C1 C1(NC(C2CN(S(CC)(=O)=O)C2)=O)CCCCN(C(C2CCCCC2(F)F)=O)C1 C12(CNC(C3C(CNC(c4ccsc4)=O)C3)=O)CCN(CC1)CC2 N1(C(c2c(C)c(O)ccc2)=O)C2CCC1CN(C(=O)CC(C)C(F)F)C2 C12(NC(CC(C)SC)=O)COC(CNC(c3cc(C(F)(F)F)ncn3)=O)(C1)C2 N1(C(C(C)C)=O)CCC(CCC2CCN(C(=O)CC3CCCCN3)CC2)CC1 c1(C(=O)NCC(CC)NC(C2CCOC2=O)=O)c[nH]nc1-c1ccnn1C N1(C(CCc2ccc(C)s2)=O)CCN(C(C2CC(F)(CO)C2)=O)CC1C1CC1 c1(OC)c(C(N2CC(NC(=O)CSC(C)C)CC(C)C2)=O)sc(C)c1Br c1(C(=O)NC(COC)C(=O)N(C)Cc2cnccn2)ccc(=N)[nH]n1 c1(CCC)ccccc1C(=O)NCCN(C(=O)CC1(C)CC1(Cl)Cl)C1CC1 n1(CC(=O)NC(C2N(C(CCC(=C)C)=O)CCC2)(C)C)ccc2ccc(F)cc12 C1(C(N(CCOCC=C)C)=O)CC(NC(=O)C(C)n2cnnn2)C(O)C1 CC1(C2CCN(C(C3CCN(C(=O)Cn4cccn4)CCO3)=O)C2)CC1 CCCC(C)(O)CC(=O)N(C1CCN(C(=O)CCOCC)C1)CCC N1(C(=O)NCc2c(O)cccc2Br)CCc2c(C(=O)O)csc2C1 C1(CC(=O)NC2(CN(C(CCOCC)=O)C)CC2)COCC(C)O1 N1(C(C2C(C(C)NC(=O)C(C)N3CC(C)C3)C2)=O)CCN(C2CC2)C(=O)C1 CC1CC(NC(C2(c3ccc(Cl)cc3)CCC2)=O)CCN1C(=O)C=CBr C(CCCC(C)(C)NC(=O)CC1CC2CC2C1)NC(c1cc(C)nnc1)=O C(=O)(CS(=O)(=O)C(C)C)NC(CCCNC(CC1C(C)=NN(C)C1=O)=O)C Cc1ncnc(O)c1CCC(=O)NC(C1CN(C(=O)Cc2nncs2)C1)C C1(C(N(CC(=O)NCC)C)=O)CCN(C(C2CCCC2OC)=O)C1CC c1(C(N2CCC(C(C(=O)NCCCC#C)(C)C)C2)=O)ccc(C#N)cn1 C1(NC(=O)CC2CCCOC2)COCCN(C(=O)Cc2ccc(Cl)cn2)C1 c1(C(N2CC3C(CNCc4cccc(OC(C)=O)c4)(C3)C2)=O)ccc(Br)c(Cl)n1 N1(C(c2c(C)c[nH]c2)=O)CCN(C(C2CCCCN2C(=O)CC(C)C)=O)CC1 CP(C)(=O)C1CCCC(NC(=NCC2CC(OC(F)F)C2)NC2CCOCC2)C1 C=CC(O)C(=O)NCC1CC(C(=O)NCCC(O)C2CCC2)C1 Cn1cc(C(=O)NC2CC2CNC(c2ccc(CCO)cc2)=O)ncc1=O C1(C(=O)NC2(C)CC(NC(=O)CC3CCCO3)C2)CC12CCCCC2 C1(CNC(C2CC(CCC)OCC2)=O)CN(C(C2CCCC2OC)=O)CCCO1 N1(C(=O)NC(C)(C)CC2CCCC2)CCN(c2n[nH]c(=N)o2)CC1 N1(C(c2c(C)oc(C)c2C)=O)CCCCC2(CCN(C(c3cc(Br)n[nH]3)=O)C2)C1 C12(C(=O)NCCCN(C(C)C)C(c3sccc3Cl)=O)CCCC1CC2 Cc1cnc(C(=O)NC2CCOC(C3CCN(C(=O)C(Cl)=CCl)CC3)C2)c(C)c1 C1(NC(C(C2(C)CC2)NC(c2c[nH]c(=NC)s2)=O)=O)CCn2cnnc2C1 c1(C(=O)OC)cnc(NC(=O)CC2CCCN2Cc2c(C)cccc2C)c(Cl)c1 CCC(C)C(O)CC(=O)NCC1(NC(=O)Cc2cn(C)cn2)CCCC1 c1(CCC(=O)N(C)CC2CCCCN2C(c2ccco2)=O)ccccc1[N+](=O)[O-] c1(NCC2CC(CC)C2)cc(Br)ccc1OC N1(C(CC2N(C(C(CN(C)C)O)=O)CC2)=O)CCC(F)C(F)C1 Cc1nnc(CCC(=O)NC2COCCC2NC(=O)C(F)(F)CC2CC2)n1C C1(CNC(c2ncn(C)n2)=O)CC(O)CN1C(C1CCC1c1ccccc1)=O N1(C(C2(C#N)CCSCC2)=O)CCC(C2CC2)(CNC(=O)C(F)(F)C(F)F)C1 c1(OC)ccnc(-c2nc(Cn3cc(C)cn3)n(C(C)C3CC3)n2)c1 C12(CNC(C3(F)CN(C(c4ncccc4Cl)=O)C3)=O)CCCN(CC1)C2 c1(CC(=O)NCC2CCN(C(=O)C(=O)C3CCCC3)C2)ccc(Cl)cn1 c1(OC)cc(NC(=O)C(C2CCCCC2)C)c(NC(C)=O)cc1OC c1(COC)ccccc1C(=O)NC1CN(C(=O)CC2(O)CCOC2)CC1OC c1(NC(C2N(C(C3(C(C)(C)C)CCC3)=O)CCC2)=O)ccc2c(c1)OCO2 C1(C)(C(N2CC(C=C)C(NC(=O)CC3NC(=O)NC3=O)C2)=O)CCCCCCC1 C1(C(=O)NCc2c(C(N(CC(Cl)Cl)C)=O)nco2)CCCCC(=O)C1 c1(C(=O)Nc2scc(C)n2)cc2c(s1)CCN(Cc1cnn(C3CC3)c1)C2 CCCCC(O)C(=O)NCC1(C(=O)N(C)CCn2cncn2)CC(C)(C)C1 C12(OCC)CC3CC(CC(C3)O1)C2.C(CCN(CCOCCO)CC)(NC)OCC CC1=C(C(=O)NC2C3CN(C(c4ccc(-n5ccnc5S)cc4)=O)CC23)CCC1 C1(CC=C)(C(=O)NCCN(C(c2ccnc(C(F)F)c2)=O)C2CC2)CCOCC1 CC1(C)CCN(C(=O)C(C2CCOCC2)F)CC1NC(c1csc(C(N)=O)n1)=O c1(C(=O)NCC2C(NC(c3nccc(CC)c3)=O)CCC2)cc(C)c(N)cc1F C#Cc1cccc(CC(N2CCC(C(C)C(=O)NCc3ccncc3)CC2)=O)c1 C1(CNC(C(C=C)(C)C)=O)CCN(C(C2CCC(CC3CCCC3)CC2)=O)C1(C)C C12(NC(c3c(C)noc3)=O)CCCC1CN(C(C1CCO1)=O)C2 C1(N(C(=O)CC2CC(F)(F)C2)C)CCC(CNC(=O)CCC2CCC(=O)N2)CC1 c1(C(N2CCC(C(N3CCOC(CCN(C)C)C3)=O)CC2)=O)ccccc1O N(C(=NCC1(NN2CC(C)CC2=O)CCCC1)NCC(=O)N(C)C)C(CC)C c1(OC)cc(OCC2(NC(=O)NCc3ccccn3)CCCCC2C)ccc1O Cc1ccc(CC(N2CCN(C(C3CCCN(C)C3)=O)CC2C(F)F)=O)c(Cl)n1 C1(CN(C(CC(C)C2CC2)=O)C)CCN(C(c2ccccc2SCC#N)=O)CC1 C1(NC(Cc2c(OC)cccc2)=O)CS(=O)(=O)CC1NC(=O)Cn1ccnn1 Cc1cccc(C(N2CCC(CCNC(C3(C)CC4(CC4)C3)=O)C2)=O)c1C Cc1nn(C)c(Cl)c1C(N1CCC(C)(CNC(=O)CCc2cnn(C)c2)CC1)=O C1(NC(c2c(C)sc(Cl)n2)=O)CCN(C(C2C3COCC23)=O)CCC1(F)F c1(C(=O)NC2(C3CN(C(C(CC)C#N)=O)C3)CC2)cc2c(=O)[nH]ccn2n1 c1(CN(C(=O)NC2C(C(N)=O)C2)Cc2ccccc2)ccccc1Br CCCC(C)CC(=O)N1CCC(C(C)(C)NC(c2cc([N+](=O)[O-])c[nH]2)=O)CC1 Cc1nc(Br)oc1C(=O)NCC1CCN(C(=O)Cc2cnn(C)c2)CC1 CCC(O)C(F)(F)C(=O)NCCC1CCCN(C(c2ccc3nn[nH]c3n2)=O)C1 c1(NC(C2CCC(NC(C(c3ccccn3)N)=O)CC2)=O)cccc(F)c1O c1(C2CC(NC(C3(CC#N)CCOC3)=O)C2)ccc(Br)cc1 c1(OC)cc(Br)cc(CN2CCNCC2C(=O)Nc2ncc(C)cc2O)c1O N1(C(C2CCCN(CC)C2)=O)CC2CCC(NC(C3CC(F)(CO)C3)=O)CC2C1 Cc1cc(NC(C2CCCC2C(=O)O)=O)ccc1NC(c1cnn(C(C)C)c1)=O C1(NC(C2CCOCCN2C(c2ns[nH]c2=O)=O)=O)CCn2ccnc2C1 CCCCC(CNC(c1nocc1C(C)C)=O)NC(C1CC=C(C)CC1)=O CC1(C)CN(C(c2cc(C(N)=O)c[nH]2)=O)CC1NC(C1CC2(CC2)CO1)=O CC1CN(C(=O)COCCOCCO)CCC1NC(=O)C(N1CCOCC1)C O(C1CCCn2c(Br)cnc21)C(C(N1C(=O)c2ccccc2C1=O)CC)=O CCCN=C(NCCc1ccsc1)NCC1CC1(F)F C1(NC(=O)C=Cc2cocn2)C2CC3CN(C(=O)CC4CSCCS4)C1C3C2 N1(C(C(C)CO)=O)CC2(CCN(C(c3ccc(F)c(C(F)F)n3)=O)CC2)C1 c1(C(C)=O)ccc(NCC(C)CNC(=O)C(C)C2CCC2)c([N+](=O)[O-])c1 N1(C(c2c(C)nc(C)s2)=O)CCC2(CCCN2C(=O)CN2CC=CC2)C1 N1(C(COCCN(C(=O)C(C)(F)C(C)(C)F)C)=O)CCCC2(CCOC2)C1 C1(C(N2CCN(c3ccccc3)CC2)=O)COCCN1C(=O)CC1CCCC1 c1(CC)ccc(N)c(C(N2CCC(NC(C3CCC4(CC3)CC4)=O)C(O)C2)=O)c1 N1(C(c2ccc(-c3c(O)ccc(C(=O)OC)c3)cc2)=O)Cc2ccc(F)cc2C1 N1(C(C(CC)n2cccn2)=O)CCC(NC(=O)Cc2cn(C)nn2)C2(CCC2)C1 N1(C(C2=CC(C)CC2)=O)C2CCC1CC(NC(c1cncc(F)c1)=O)C2 CCCCC(C)N=c1[nH]c(N(CCCOc2ccccc2)C)nc2c1CCC2 c1(C(=O)OCc2n(C)ncn2)ccc(OCCNC(C2C(F)(F)C23CC3)=O)cc1 C1(NC(Cn2c(C)c(Cl)cn2)=O)CN(C(=O)CC2CC(F)(F)C2)CC12CC2 Clc1cc(C2CC2)nc(=NCC2CCc3c[nH]nc3C2)[nH]1 c1(C(C(=O)OC)OC(C2CC(C(=O)N(C)C)C2)=O)cc(Cl)ccc1Cl C1(NC(c2nc(Cl)ccc2F)=O)CCN(C(c2cnsc2)=O)C12CCC2 c1(C(=O)NC2CN(C(CSCC#C)=O)C(C)C2)ccc(C)cc1OC N1(C(c2c(C)noc2C(C)C)=O)CCCCC(NC(c2cc(C(N)=O)co2)=O)C1 CC1(C)CCN(CC(N2CCCCC2CCNC(C2C3COCC23)=O)=O)C1 C1(CNC(C(=O)NCC)=O)CC(NC(c2sc(C)cc2C)=O)C1(C)C c1(CC)nc(C)c(C(=O)NCC(C(C)(C)C)NC(=O)CC2CC(=O)C2)c(C)n1 C12(C(N3CC(CCNC(C=CC(=O)OCC)=O)C(C)C3)=O)CC(CO)(C1)OC2C N1(Cc2cn(CCC)nc2)CC(NC(=O)Cc2noc(C)n2)C(C#N)C1 C#CCC(CC(=O)OC)NC(=O)NCC(c1cnn[nH]1)N1CCCC1 N1(C(C(C)OCC=C)=O)CCOCC1C(=O)NC1CC(N2CCC2)C1 c1(C2(C(=O)NC3CCN(C(COCCCC)=O)C3)CC2)ccc(F)cn1 N1(C(c2c(C)ocn2)=O)CC(C(=O)N2CC(O)CO2)CCC1(C)C C1(N(C)C)CC(NC(c2conc2CNC(=O)C=Cc2ccncn2)=O)C1(C)C c1(C(N(CCCCCNC(C(C2CCC2)OCC)=O)C)=O)cccn2nnnc12 N1(C(c2cc(CC)no2)=O)C(CNC(c2ccc(C3CC3)o2)=O)CC2CCCC12 C1(C(N2CC3(CN(Cc4c(C)cccn4)C3)C2)=O)Cc2ccccc2CN1C N1(C(c2nc(C)oc2)=O)CCCC2(C1)CN(C(c1csc(CC(F)(F)F)n1)=O)C2 c1(C(=O)NC2CC(C(N(CCn3ncc(C)c3)C)=O)OCC2)ccc(C)c(C)c1 CCCCC(CCCC)CC(CC)N1CCC(C)(C(=O)OC)C1 Cc1ccc(C)c(C(N2CCOCCC2C(N2CCC(O)(CO)C2)=O)=O)n1 C1(C(C)C)CN(C(=O)C(N2CCCCCC2)C)CCCN1C(c1cnsn1)=O N1(C(c2c(N)ccc(Cl)c2)=O)CCC2(CCCCC2NC(=O)C(F)CC2CC2)CC1 c1(C(=O)NC(CC(C)NC(c2ncc(OC)nc2)=O)C)ncnc2ccsc12 c1(C(N2C(C(=O)NOCCCCF)CCC(O)C2)=O)c[nH]c2cnccc12 c1(C(=O)NC2C(C(=O)OCC)CCC=CCC2)cc2cc(Br)ccc2o1 CC1(C)CCN(C(=O)CC(=O)NC2CCCCC2F)C1.C12CCCN(C1)C2=O c1(C(N2CCC(OC)(CNC(=O)CC(F)F)C2)=O)cccc(S(N)(=O)=O)c1C Cn1ncc(CNC(C2CCC(NC(c3cccc(O)c3)=O)C2)=O)c1O c1(C(=O)NCC2(CNC(CNS(CCCC)(=O)=O)=O)CC2)nccc2nn[nH]c12 c1(C(=O)NC(C2CCOC2)CNC(CN(C)C2CC2)=O)cc2ccccc2n1C C(=O)(C(C)(C)n1cc(Cl)cn1)NCC(C)NC(=O)CC(c1ccccc1)C1CC1 c1(C(=O)NCC2CN(C(C3C(C)(C)CO3)=O)C2)c(F)ccnc1Cl n1(Cc2nc(N(C3CCc4nnnn4C3)C(C)=O)sc2)cnc2c(C)cccc2c1=O c1(C(=O)OC)c(Cl)cccc1S(=O)(=O)NC(C1CCCCO1)C C12(NC(c3cc(C(F)(F)F)ncn3)=O)CCCC1CN(C(c1csc(Cl)c1)=O)C2 C(CNC(C1CCCN(C(c2nc(C)sc2C)=O)C1)=O)(CC(C)C)OC C(=O)(C=CSc1nc[nH]n1)NC1C(CNC(=O)Cc2ccco2)C1 c1(C(=O)NCC(CC(C)C)NC(C2(N(C)C)CCC2)=O)ccc(O)c(F)c1F Cc1ccc(C(=O)NC2CC(O)CN(C(=O)C=Cc3cccc(F)c3)C2)c(C)c1 c1(C(N2C(CN(C(C=CCCC)=O)C)COCC2)=O)cc2c(Br)cccc2[nH]1 S(=O)(=O)(c1ccc(C(=O)NC(C2CN(C(C3(C(C)C)CCC3)=O)C2)C)o1)NC CS(=O)(=O)C1CC2(C1)CN(C(C1CCCC3(C1)N=N3)=O)C2 C1(NC(C2C(C)CCCC2)=O)CCN(C(C2CC23CC(O)C3)=O)C(C)C1 C1(NC(c2nc(C)oc2)=O)CCc2nc(NC(c3cncc(O)c3)=O)sc2C1 n1(CC)cc(CC(=O)NC2(COC)CN(C(=O)CCCOC(C)C)C2)cn1 Cc1csc2nc(Cc3nc(-c4ccc(C(C)C)cc4)nn3C3CCOC3)cn12 C1(NC(c2c(COC)ncs2)=O)CC(NC(c2nocc2C(C)(C)C)=O)CC1O Cc1ccccc1CC(=O)N(C(C)C(=O)NC1(C)CCOC1C)C1CC1 CCCN(OC)C(=O)CC(C)NC(=O)C1=NOC(C)C1C C(N=c1ccn(CC2CCOC2)[nH]1)(c1cccc(CC)n1)c1nnnn1C C1(C(=O)NC(CC#C)CC)CC2CC2N1C(C1CS(=O)(=O)C1)=O C1(C(N2CCN(C3CCCN(C(C4CCCC4)=O)C3)CC2)=O)CC1C1CCCC1 C1(CC(=O)N(C2(CC(=O)NCC(C)CO)CC2)C)CCN(C)CC1 c1(OC)nc(Br)ccc1CNCc1cccc(C(N2CCC(Br)C2)=O)c1 c1(C(=O)NCCC(=O)NCCNC(C2CCC3CCC23)=O)ccc(Cl)cc1 c1(NC)cccc(C(N2CC(C(O)C(=O)NCC(C3CCCCC3)O)C2)=O)n1 N1(C(CCS(=O)(=O)NC)=O)CCOC2(CCN(C(C3CCCC3OC)=O)CC2)C1 C(=O)(C1COc2ccc([N+](=O)[O-])cc21)N1CC(NC(CN(C)CCO)=O)C(O)C1 C1(c2cccs2)(C(=O)OC)CC2(CCC2)C1.C12(O)CCN(C1)c1nnnn1C2 C12(CNC(c3c(CC)noc3)=O)CN(C(=O)C(C)OC)CC1(C(F)(F)F)C2 C12(C(N3C(C(=O)OC)C=CC3)=O)COC(C1)C(NC(c1cnccc1C)=O)C2 N1(C(CCC)=O)CCC2(NC(=O)Cc3ccc(Cl)cc3C)CCCCCC12 c1(OC)ccc2c(c1)C(O)(CNc1ncc(Br)cc1C#N)CC2 C(=O)(C(CCC)C(C)C)N(CCC(N1CC2(CCC2O)C1)=O)CC=C c1(C(N(CCCNC(C2CC2C(F)F)=O)C(C)C)=O)cc(Cl)c(N)cc1F C1(C(=O)NC(C2CCCC2)CO)CCCCCN1C(=O)Cc1ccsn1 C1(NC(C(C(C)(C)C)O)=O)CC2CCC1CN(C(c1ccc(O)c(N)n1)=O)C2 c1(CCC(N2CC3CN(C(C4CC4(Cl)Cl)=O)CC3C2)=O)nc2cnccc2[nH]1 C#CCC(CC(=O)N1CCOC(C#N)C1)NC(=O)CCC(C)SC C1(NC(c2cc(Cl)c[nH]2)=O)CC2CC1CN2C(=O)Cc1csc(C2CC2)n1 c1(C(=O)NCC(C(C)(C)C)NC(=O)CC2CCCO2)cc2ccccc2o1 C(=O)(C1(C)CCOc2ccccc21)N1C(CCNC(CCC=C)=O)CSCC1 C(c1c(F)cccc1F)=CC(=O)N(c1c(C)ccc(C)c1)C c1(C(=O)NC(CCCC)CNC(C2CC2CCC)=O)scc2c1OCCO2 C1(Sc2ccccc2)CCCCC1CCNC(CCSCC(=O)OC)=O C1(N(C(=O)Cc2csnn2)C)CCC(NC(c2coc(C(F)F)c2)=O)CC1 c1(CC)cnsc1C(=O)NC(C1CCCCC1)CNC(c1nsnc1O)=O CC1(C)CN(C(=O)C2=NNC(C(F)(F)F)C2)CCC1NC(c1ncccc1O)=O c1(C(=O)NC(CNC(C(C(C)(C)C)O)=O)CO)cccc2ccncc12 c1(C(N(C)CC2(NC(CC(C)c3ccncc3)=O)CC2)=O)cnc(C(N)=O)cn1 N1(C(Cc2c(C)nc[nH]2)=O)CC2N(C(c3cnc(C(C)(C)C)[nH]3)=O)CCC2(C)C1 C(CSC)(C(=O)NC1CCN(C(N)=O)C1)NC(CCOC)=O c1(C(N)=O)cccc(C(N2CC=CC2CNC(C2(O)CCSC2)=O)=O)c1 c1(OC)ncc(C(N2CCN(c3ccc(-c4nn[nH]n4)cn3)CC2)=O)nc1C N1(C(C=C(C)C2CC2)=O)CCN(C(=O)CCc2nnc(C(C)C)o2)CCC1C CCCCC(O)C(=O)N(CCNC(=O)CC1CCOC1=O)CCc1ccccc1 c1(CN2CC(CNC(c3ccc(Br)cc3O)=O)C2)cc(Cl)ccc1F C1(CC(=O)NC2CC(NC(=O)CNc3nccs3)C2)CC2CCC1O2 n1(CCC(=O)NC2C(NC(C(C)NC(C)=O)=O)CC2)cnc2c(cnn2C)c1=O CC(C)C(O)CC(=O)NCC(O)CN(C(=O)Cn1ncc(O)nc1=O)C c1(C(=O)NC(CC)CN(C(=O)Cn2nccc2C)CC)cc2ccsc2c(O)n1 Cn1nnc(C(=O)NCC(CO)NC(=O)C(=C2CCCCC2)F)c1N C1(NC(C2CCC(NC(c3c(CC)cno3)=O)C2)=O)CC(C)(C)C1OC N1(C(=O)Cn2cc(CO)nn2)CCN(C(=O)CC2CCCS2(=O)=O)C(C2CC2)C1 CN1CCCC(CCC(=O)NCCOC2CCN(C(c3cnns3)=O)CC2)C1 C(=O)(CCCCCCNC(=O)CC1CCCC(=O)N1)N1C(C)(C(=O)OC)CCC1 c1(C(=O)NC2CCN(C(C(C)OCC#C)=O)CC2)cc(OC)ccc1C N1(C(C(CC=C)(C)C)=O)CCCC(C2CCN(C(C3CCCCCC3)=O)C2)C1 c1(C(=O)NCCCOCCC(=O)NCC2(O)CCC(C)C2)cc2ccccc2o1 C1(C)(C(C)C)CCN(C(=O)C(C2(O)CCC2)NC(=O)CC23CCCC2C3)CC1 C(=O)(C1Cc2c(Cl)cccc21)N1C(C)(CNC(=O)CN2CCSCC2)CCC1 C(CCOC)(C(=O)N(C1CCCC1)C)NC(C(C)=C(CC)C)=O C1(NC(c2cccs2)=O)CC2CC1CN2C(c1ccnc(C(F)F)c1)=O N1(C(C)C)N=C(C(=O)N2CCC2CNC(C2CC3(C(OC)CC3)C2)=O)CCC1=O Cc1c(-n2cc(CC3CCCN(C(C4(O)CCOCC4)=O)C3)nn2)cnn1C O=C(C1=CC2(CCOC2)C1)N1CCC2C(C1)CN2C(=O)C=Cc1cccs1 Cc1ccc2ccc(C(=O)NC3CCOC3=O)nc2c1.C12CCC(CC1)CN2C N1(C(C2C(=C)C2)=O)CC(O)CC1(C)C(N1CCC1C(=O)N(C)C)=O c1(SCC)cc(C(N2CCCC(NC(=O)C(C)(C)CSC)C2)=O)ccn1 c1(CC)nccc(N2CCC(CNC(c3cnn(C)c3N)=O)(OC)C2)n1 N1(C(C(c2c(OC)cccc2)C)=O)CCN(C(=O)C(CO)N(C)C)C(C(C)C)C1 C1(C(=O)NCCN(CC)CC)CCN(CCC(=O)Nc2ccc(C)cc2)CC1O C#CC1(O)CC(C(=O)NC(CCF)C(=O)NCCNC(=O)CO)C1 c1(C(=O)NC2CC(C)N(C(=O)COC3CCC3)CC2)cnc2c(c1)NC(=O)CS2 c1(OCC(=O)NCCNC(C2(CC)CC2C)=O)c(Cl)cc(Cl)cc1Cl C1(C(=O)Nc2c(C)[nH]nc2Cl)CN(Cc2ccc(-n3cncn3)cc2)CCC1O C(=O)(C(C(C)C)n1cnnn1)NC1CC(C)(NC(c2c(C)nc[nH]2)=O)C1 C(=O)(C1=NOC(C)(C)C1)N1CCC(C(N2CCC(OCC=C)C2)=O)C12CC2 C(=O)(CCCCCCCO)N1CC2CCN(C(c3cc(O)ncn3)=O)C2C1 C1(NC(c2c(C)n(C(C)C)nc2)=O)CC2CN(C(C3CC(=O)NC(=O)C3)=O)CC12 C=CC1(CO)CCN(C(=O)Nc2ncccc2Cl)CC1 N1(C(c2occc2CC)C(=O)NCCCCCC)CCC(C2CC(F)(F)C2)C1 N1(C(CSCC#C)=O)CCC2CCCC12CNC(C1(COCC)CC1)=O C1(C(=O)NCCCOCCNC(C2(N(C)C)CCC2)=O)CCN(C)C(=O)C1 c1(C2CCCN(C(=O)NC3CCCC(F)C3)C2)ccc2cccnc2n1 N1(C(c2cc(C)n(C)c2)=O)CCC2(CC1)C(NC(c1ccnnc1)=O)CS2(=O)=O C#CCCC(C(=O)NCC1CN2CCC1CC2)NC(c1ncsc1NC)=O c1(C2(CCNC(C3CCCN3)=O)CC2)cccc(C(F)F)c1 CCC(CC)C(C(=O)NC1CC2CC1CN(C(=O)CSCC(F)(F)F)C2)OC CC(C)C(F)C(=O)N(C1CCN(C(C2(C(c3ccccc3)=O)CC2)=O)C1)CCO N1(C(c2ccc(Cl)nc2F)=O)CCc2cc(-c3cc(CO)ccn3)ccc2C1 C1(CNC(C=C(C)C(C)(C)C)=O)CN(C(=O)CO)C2CC12 C1(NC(c2cnc(C3CCC3)s2)=O)CCC(F)(CNC(c2ccccc2Cl)=O)C1 N1(C(=O)CCCn2cc(-c3ccncc3)nn2)CCC2(CCCCC2)C(O)C1 c1(OC(C(=O)NC(C2CN(C(CCCC)=O)C2)C)C)ccc(Cl)cc1C c1(-c2n(CCOC)ccn2)ccc(S(=O)(=O)NC2COC23CCNCC3)cc1 c1(CC(=O)NC2(CN(C(CC3ON=C(C)C3)=O)C)CC2)cnn2c1OCCC2 C=C(C)CCCC(=O)N1CC(CNC(C2CC(C)C2(C)C)=O)(OC)C1 C12(C(=O)NCCCCC(C)NC(C(C)O)=O)CC3CC(C)(C1)CC(C)(C3)C2 n1(CC(C)C)ccc(=NC(=O)C2(C)CCCN(C(c3cnn4c3OCC4)=O)C2)[nH]1 CCC(CN(C)C)C(=O)N1CC2CC1(C(=O)NCC(F)(F)Cl)C2 C1(CNC(C(C)CSc2ccccc2)=O)CC(C2CNC2)C1 C1(CNC(CCOCC)=O)CCCCCN1C(C1CCCN1C)=O C(CC(C)(C)NC(=O)C(C)n1cncn1)N(C(COC(C)C)=O)C C12(CNC(C3CC(n4cc(-c5cncc(C)c5)nn4)C3)=O)CC1COC21CCC1 CC1CC(NC(=O)CSc2cccc(Cl)c2)CCN1C(=O)C(Cl)=CCl C1(NC(=O)Cc2cscn2)CN(C(C2CCCCC(F)(F)C2)=O)C2CCCC12 C(=O)(C(C)C(=O)NC(c1nc(C(N2CC(CCO)C2)=O)co1)C)OC C#CCC(CC(F)F)C(=O)N1CCCC1CCC(=O)N1CC(c2cc(O)n[nH]2)C1 c1(SCC)cccnc1C(=O)NC1CC(C(=O)NCCCCCF)C1 N1(C(C2(C)CC2)=O)C2CCC1CN(C(=O)Cc1csc(C3CC3)n1)CC2 N1(C(CC2CN(C(C)=O)C2)=O)CCCC(CNC(=O)CSc2cn[nH]c2)C1 C1(F)(C(N2CCC(NC(C3(O)CCC(CCC)CC3)=O)C2)=O)CCC(F)(F)CC1 C12(COC)CN(C(=O)Cc3cnn(C)c3)C(CNC(C3(C)CC(F)(F)C3)=O)(C1)C2 c1(C(N2CCC(CCNC(CCC#C)=O)CC2)=O)cc(F)c(Br)cc1Cl C1(C(N(CC(CCC)C)C)=O)CC2CC1CN(C(C1(Cl)CCC1)=O)C2 C1(C)(C(=O)NCC(=C)CCNC(c2ccns2)=O)CCOC(C)C1 c1(C(N2CC3N(C(c4ccc(C)nc4)=O)C3C2)=O)ccc(F)c(F)c1F N1(C(CSCC#C)=O)CCCC(NC(c2cc(SC)c(C)o2)=O)C1C N1(C(c2cocn2)=O)CC2CCC1C1CN(C(c3ccc(C4CC4)cc3)=O)CC21 N1(C(CCCC#C)=O)CCC(NC(=O)C2=CCCC2)C12CCCC2 CC1(C)C(CC(=O)NCCC2CCN(C(c3cccnc3S)=O)CC2)CC1O C(C(=O)NC(c1ccccc1)CNC(=O)C(CCO)N(C)C)(C(C)C)OCC N1(C(C2C(C)CCC2)=O)CC=C(CCNC(c2ccc(SC(F)(F)F)[nH]2)=O)CC1 c1(CC)nc2sc(C)cn2c1C(=O)NC1CN(C(=O)Cc2n[nH]c(C)n2)CC1C N1(C(=O)OC(C)(C)C)CCCC(C)(CNCc2ncc(Cl)s2)C1 c1(C(N(CC(C)NC(C(c2ccccc2)C)=O)C)=O)c(F)ccnc1Cl c1(C(N2CCN(C(CCC(C)OC)=O)CC2CCO)=O)ccn2c(C)cnc2c1 CCC(CC(=O)N1CC(C)CCC1C(=O)NCc1cnn(C)c1OC)C(C)(C)C C1(NC(C2C(C)CN2C(c2cnn(CCF)c2)=O)=O)CC(C2CCCC2)C1 c1(C(N2C(COC)(CNC(=O)C=CC3CCOC3)CCC2)=O)ccc(C)c(O)n1 C(=O)(CC(C)P(C)(C)=O)NCCOCC(N1CC(O)(C(C)C)C1)=O c1(N2CCN(C)C(CNC(=O)CCC3CCCO3)C2)ncc2ccsc2n1 c1(C(=O)NCC2C(C)CCN2C(c2ccoc2Br)=O)cc2nnn(C)c2s1 C1(CNC(C(CC)F)=O)CC2(CCN(C(=O)CC3CCCC(=O)N3)C2)CO1 C1(NC2CC(C(C)C)OCC2)CC2CC1CC2F c1(CC)ccc(F)c(C(=O)NC2COCC2NC(=O)C=CC(=O)NCCOC)c1 C1(NC(C(CCC)NC(=O)CCc2ncnn2C)=O)Cc2cscc2C1 c1(NC(=O)NCC(n2cnc(C#N)n2)C)nc(N2CCCC2)ncc1Cl c1(C(N(CCCNC(CCOCCOCC)=O)C)=O)conc1C C(=O)(C(C(C)C)c1ccn(C)n1)N(CC(C)NC(c1ccc(C(C)=O)o1)=O)CC CCC(C)C(CC(=O)NC1(C2CCCO2)CC1)NC(=O)CS(C)(=O)=O N(C1COc2cccc(Cl)c21)C(c1cnc(Br)c(Cl)c1)=O c1(C(=O)N(C)C)ccc(-c2cccs2)o1.O1NC(=O)NCC(C2CC2)N(C)C(=O)C1 C1(CNC(c2n(CC)cc(Cl)c2)=O)C(C2CC2)CCN1C(c1cnnc(Cl)c1)=O N1(CC(=O)NCC2CCCN(C(c3cccnc3O)=O)C2)CC2C=CC1C2 CCCCC(=O)NC1(C2CCCN2C(c2cc(-c3csc(=N)[nH]3)c[nH]2)=O)CC1 C(=O)(C(C)C(O)CCCC)NCC1(C(=O)Nc2ccc(C)c(C#N)c2)CC(=C)C1 C(=O)(CC(C)(F)F)NCC1(C(=O)NCC(=O)NCC(C)N2CCC2)CCC1 N1(C(CC=CCC)=O)CCC(CO)(NC(c2nc(C(F)(F)F)cn2C)=O)CC1 CC1(NC(c2coc(Br)n2)=O)CCCN(C(=O)CC2(c3ccon3)CCC2)C1 C1(C)(CC)CCCN(C(C2CN(C(=O)Cc3ccc(Cl)cc3)CC2F)=O)C1 c1(C(N2C(C)(C)C(NC(=O)CCC(=O)NC=O)CC2)=O)ccc2c(c1)COC2 c1(COC)ccnc(C(N2CC3CC2C3NC(C2CCOC2C)=O)=O)c1 Cc1cc(C(=O)N(CCN(C)C(c2snnc2C2CC2)=O)C(C)C)nn1C(C)C c1(OC)cc(C(N2CCN(C)C(CNC(=O)CN3CCCC3)C2)=O)cc(Cl)c1 CCCCC(CNC(=O)CCCC1CCCO1)NC(C1CSCC(=O)N1)=O C1(NC(c2c(C)c(F)ccc2)=O)CN(c2ncc(I)cn2)CCC12CCOCC2 c1(C(=O)NCC(CC(C)C)NC(Cc2c(C)n[nH]c2C)=O)coc(S(N)(=O)=O)c1 N1(C(C23C(C(N)=O)(CCC2)C3)=O)CC2=C(C1)CN(C(C1(F)CCS(=O)(=O)C1)=O)C2 N1(C(C=Cc2occ(C)n2)=O)CCOC2CN(C(=O)C=Cc3cnn(C)c3)CC12 c1(C(N2CCC(CN(C)C(C3(O)CCSC3)=O)C2)=O)cc2cc(F)ccc2[nH]1 CC(=O)CCCC(=O)NCC1CCN(C(C2C3(CC3)C23CC3)=O)C12CC2 CCC(C#N)(CC)C(=O)NCCN(C(=O)C(C)C=Cc1ccccc1)CC(C)O C(=O)(CCCC(F)(F)F)NC1CCC(N(C(C2C(C)CC2C)=O)C)CC1 N1(C(C2(CC(=O)OCC)CCCC2)=O)CC(C(=O)NCc2ocnc2C)C(C)C1 C(C1=CCN(C(=O)CC2CCC(F)(F)CO2)CC1)NC(c1c(C)nns1)=O Cc1cc2cc(C(=O)NC3C4CCC3N(C(C3CCSC3)=O)C4)c(Cl)cc2[nH]1 Cc1ccc(CC(=O)NCC2(NC(C3C=CCC3)=O)CC2)cc1 CC1CCCN(C(c2cnn(C)c2F)=O)C1CNC(C1CCC(C(N)=O)CC1)=O C(CCCC(CO)NC(c1cc(C2CC2)ccn1)=O)NC(CC(=C)C)=O S(=O)(=O)(c1cccc(C(=O)O)c1C)NC(C(CC)N)c1ccccc1 Cc1cnc(C(=O)N(C(C)CN(C)C(c2nc(C(C)(C)C)no2)=O)C)c(C)c1 S(=O)(=O)(c1nccs1)N1C(C(=O)NC2CS(=O)(=O)C2)CCCC1 N1(C(c2c(OC)n[nH]c2)=O)CCN(C(c2cc(Cl)c(Cl)n2C)=O)C(C2CCC2)C1 CCN=c1[nH]c(C(=O)N(CCC(C(C)(C)C)NC(c2cccnc2)=O)C)cs1 c1(C(N2CCCNCC2C(C)C)C(=O)NC)c[nH]c2cnccc12 C1(NC(=O)Cc2ccoc2)CCN(C(=O)CCc2ccncn2)CC1CO c1(OCC(=O)NCC(O)CCc2ccccc2)ccccc1Br c1(NC(N(CCCNC(C=C(CC)C)=O)C)=O)ccccc1.C1(=O)CCN1 c1(C(=O)OCC)ccc(C(=O)NCCCC(C)NC(=O)Cn2cc(C)cn2)cc1 C1(CN2C(c3ccc(F)cc3Cl)CCCC2)CCC2(CCCC2)C1 C1(C#N)(C(=O)NCC(C)N(C(C(C)Cc2ccccn2)=O)C)CC2(CCC2)C1 N1(C(C2CCC(OC)CC2)=O)CCCC(NC(c2cccnc2)=O)C1C C(=O)(C1=NOC(C)(C)C1)N1CC(C2C(C(N(c3cccc(O)c3)CC)=O)C2)C1 c1(C(=O)NC(COC)CNC(=O)C(CSC)OC)cnc(C)c(C#N)c1 c1(C(C)NC(=O)NC(C#C)CC2CCOC2)nnc2ccccn12 C(=O)(CS(=O)(=O)CC(=O)NCCCNC(=O)CCc1cc(C)n(C)n1)OC c1(C2(C(=O)NCCCNC(C(C)C3CCCC3)=O)CC2)cccc(F)c1 C1(C2CCCN(C(=O)C(C)(C)C(F)F)C2)(NC(c2c(C)[nH]nc2C(F)F)=O)CC1 C1(C(=O)NC2CCCN(C(=O)C=CC3CCCO3)CC2)Cc2cc(Cl)ccc2O1 c1(C(=O)NC(CCOC)CNC(=O)C(CO)N(C)C)cc([N+](=O)[O-])cn1C C12(CNC(CC3CN(C)C3)=O)CCC(C1)N(C(=O)CCn1cc(Cl)cn1)C2 C1(NC(C2CCC2)=O)CN(C(=O)CCC(F)(F)F)C2CCCC12 Cc1cc(CN2CCC(O)(C(=O)NCc3ccc(Br)cn3)C2)ccc1[N+](=O)[O-] c1(NC(CSCC=C)=O)ccccc1CNC(=O)C(=O)NCCOC N1(C(CC2OCC(C)(C)C2)=O)CC(O)CC1(C)C(=O)NC1CCCC(O)C1O CC(C)C(O)C(=O)NCCCC(C)(C)NC(=O)C(C)Oc1ccc(C(N)=O)cc1 c1(SC)nc(Cl)c(Br)c(=NC(=O)c2cc(Cl)cc3[nH]ncc23)[nH]1 c1(C(N2CCCC(O)CC2)C(=O)NC2COC2)noc2c1CCC2 c1(CCC)c(C(=O)NC2(C)CC(NC(C3CCCCC3OC)=O)C2)nnn1C CCC(C)CCC(=O)NCC1CCC1NC(=O)Cc1coc(C(F)F)n1 C(C(F)F)(C(C)(C)C)NC(CC(C1CC1)NC(C1C(C)CCO1)=O)=O N1(C(C(=O)NC(C)C)=O)CC2(C1)CN(C(c1occc1Cl)=O)CCO2 Cc1ccc(CC(N2CCC(O)(CN(C(=O)C(F)(F)CC3CC3)C)C2)=O)cc1C C1(C)(C(N2CC(NC(=O)OC(C)(C)C)C2)=O)CCNC1=O C(=O)(CCS(C)(=O)=O)NCC(c1cccc(N(C)C)c1)NC(c1cnnn1C)=O N1(C(C)C)CC(C(=O)NC2CC(NC(=O)C(c3ccc(F)cn3)(F)F)C2)CC1=O C=C1CCN(C(=O)C(C2CC2)C2CC2)C(C(=O)N(C)Cc2ccccc2C)C1 C1(C)(C(=O)OC)CCN(C(C2(N(C(=O)C(=O)Nc3ncc[nH]3)C)CC2)=O)C1 c1(C(N2CCN(C(C3N=C(C)SC3)=O)C(C)C2)=O)noc2c1CCCCC2 C1(NC(=O)COCC2CC2)(CO)CCN(C(c2cnc(C(F)(F)F)s2)=O)C1 C1(NC(c2c(CC)nns2)=O)CCN(CCOC2CCCCC2)CC1C c1(CC(=O)NC2CCN(C(Cc3ncc(C)s3)=O)C(C)C2)nnc2n1CCOC2 CCCS(=O)(=O)C(C)C(=O)NCCCN(C(c1ccc(C)nc1O)=O)C1CC1 O=C(N=c1c(Cl)c[nH]cc1Br)C1(c2cccc(-c3ccc(F)c(F)c3)c2)CC1 CCC(C(=O)N1CCC(C(=O)NC(C)C(=O)OC(C)C)C(C)C1)C(C)C c1(SCC(=O)NC2(CO)CN(C(C(c3cc(C)sc3)(F)F)=O)C2)cccc(Cl)c1 CC1(C)C(NC(=O)CNc2cccc(C#N)c2)CCN1C(C1C=CCC1)=O C(=O)(C(C)C(C)NC(c1cc(Cl)no1)=O)NCCC(=O)NC(C)C c1(C(=O)NCCSC)csc2c1CCN(C(=O)C(=O)c1ccco1)C2 C(CCCCC(=O)NC1(CC(=O)NCCC2CC=CCC2)CCC1)=CCCC N1(C(CSCCC)=O)Cc2ccccc2C1CNC(=O)C(C)CC(F)F N1(CCNC(C)(C)C#N)CCC12CCCC(C)(C)C2 FC1(F)CCC(N=c2ccnc(NCCC3CCCO3)[nH]2)CC1 N1(C(=O)NCCOCCOCCOC)CC2(C1)CN(C(=O)CC1=CCCC1)CCO2 c1(C(C(=O)NCC(C)(C2CCC2)OC)NC(=O)OC(C)(C)C)cccnc1 C1(n2cnnn2)(CC(=O)N(CC2ON=C(C)C2)CC2CC2)CCCCC1 N1(C(C2C(CC)CCC2)=O)CC2CN(C(C3C4CC5C(C4)C35)=O)CC2C1 c12cccc(c1N)OC(=O)c1cc-2[nH]n1.C1(CCC)CN(OC(F)F)CC1CO c1(CC)cnc(O)c(C(=O)NC(CO)CCCCNC(=O)CCCc2ccsc2)c1 C1(C(=O)NCCc2scc(C)n2)CCCN(C(c2ccn(C)n2)=O)C1C N1(C(CCC(CC)C)=O)CCC2CN(C(c3cn4ccnc4s3)=O)CC2C1 CCC(CC)C(=O)NC(C)CCNC(=O)Cc1ccc(I)cc1 C(=O)(C(C)CC(C)C)N(CC(C)N(C(CCNS(CC)(=O)=O)=O)C)C C(=O)(C1=CC2(CCOC2)C1)N1C(C(=O)NC(c2cncs2)C)(CC)CCC1 C1(NC(C(C=C)(F)F)=O)CCN(C(=O)CC(C)c2ccco2)CC1O CCCC(C)(O)C(=O)NCC1CC(C(=O)NCCOC(F)F)CO1 CC1CCN(C(c2nccc(Cl)c2Cl)=O)CC1NC(C1CCOCC1)=O CCCCCC(CC)C(=O)NCC1(C(=O)N(C2CCCC2C#N)C)CCCC1 C(CNC(=O)CCCCCN(C)C)(C(C)C(C)C)NC(c1ccc(CCC)s1)=O C1(N(CCCCO)C(C)=O)CCN(C(=O)Cc2csc(C)n2)C12CC2 N1(C(CCOC(C)=O)=O)C2CCC1C(CNC(c1cc(CO)c(C)o1)=O)C2 c1(NC2(CCCNC(C(C)Sc3ccccn3)=O)CC2)ccc(C#N)cn1 N1(C(CCc2cc(C)c(Cl)nc2)=O)CCC2(C1)CN(C(c1ccncc1Cl)=O)C2 Cc1cc(N(C)Cc2ccc(Br)o2)nc(NC2CCCC(CC(N)=O)C2)n1 c1(OC)ccc(C(O)C(=O)NCCCCN(C)C(C2(N(C)C)CC2)=O)cc1 c1(C(N2CCC(C(C)NC(=O)CCC3CCCN3C)C2)=O)ccccc1C(F)F c1(C(C(=O)OCC#CCOC)NC(=O)OC(C)(C)C)ccc(Cl)cc1Cl C(=O)(C(O)CCc1ccccc1)N1CC(C(C)NC(=O)CCN2CCC2)C1 C1(CNC(C2CCC3(C2)CC3(F)F)=O)CC2(CCN(C(=O)CC3CC3)CC2)CO1 C1(OCCNC(C(CC)N(C)C)=O)CCN(C(=O)COc2ccc(C)cc2)CC1 C1(C(=O)NC2CCN(C(CC=CC)=O)C2)CC12CCSCC2 c1(C(=O)NCC(C)CNC(c2cc(C3CC3)cs2)=O)cccc2ccc(O)nc12 C(=O)(C(C)(C)C(N)=O)NCC1C(NC(CC(CC)C)=O)CCC1 C(=O)(C(F)(F)C1=CCOCC1)N1C2CC(CC(NC(CCNC(=O)NC)=O)C2)C1 Cc1cccc(C(N2CC(O)CC2C(=O)N(C(C)C(C)(C)O)C)=O)c1N C1(CNC(CN(C)C(N)=O)=O)CN(C(=O)CCC(=O)c2cccnc2)CCO1 C1(C(=O)NCC(CN(C)C(c2cnccc2C#N)=O)(C)C)CCN2CCCC2C1 C1(C(=O)Nc2ncccc2C2CC2)CC(F)CN(C(c2cncc(F)c2)=O)C1 N1(C(CN(C(c2cnc(O)o2)=O)CC)=O)CCC(CO)C(O)C1 c1(NC2CC3CN(C(=O)C4=CCCOC4)CC32)ncc2ccnc-2[nH]1 c1(-n2c(C(=O)NC3CN(C(CC4C(C)C4)=O)C3)cnn2)cc(Cl)ccc1Cl N1(C(CC2CCC(C)(C)O2)=O)CCC2(CCCCN(C(c3cn[nH]c3)=O)C2)C1 N(C(=NCC(F)(F)c1ccc(C)cc1)NCC1CCOC1)C(C)CC(F)F CCCCCCCC(F)C(=O)NC(CN(C(C1C(C)(C)C1(F)F)=O)CC)CC c1(NC(C(N2C(COC)CCC2)c2sncc2C)=O)cccc([N+](=O)[O-])c1 CCCCCC(=O)NC1CCCN(C(=O)CC2(C(F)(F)F)CNC(=O)C2)C1 O=C(CCCCNC(C1CCC(C2CC2)C1)=O)NOCCN1CCCC1=O C(=O)(CC(C)(C)C(F)F)NC(C)CCCCNC(=O)Cn1cccn1 C1(CCOC)(NC(=O)C(C)OC)CCN(C(C2CCC2COC)=O)C1 C(=O)(C(C)CC(N)=O)NCCCCC(C)NC(c1ccc(-c2ccco2)o1)=O N1(C(COCCC#C)=O)CCC2C(CCCN2C(=O)CC2CSC2)C1 N1(C(c2ccc(OC)cc2Cl)C(=O)NCC(F)F)c2ccc(Br)cc2CC1C N1(c2nccc(C(=O)OC)n2)CCC2(CC1)CC(OC(C)(C)C)C2 C(=O)(C#CC1CCCC1)NCCC(C)N(C)C(c1ccc(C2CCCO2)[nH]1)=O N1(C(c2nn(CC)nc2Br)C(=O)NCc2ccccc2)CCC(F)(F)C(C#N)C1 CC1(C(N2CCN(C(c3ccns3)=O)C(C3CCCC3)C2)=O)CC2CCC1O2 Cc1cccc(OCC(=O)NC(C)(CNC(=O)CC23CC(C2)C3)CO)c1 c1(C(N2CCOCC2C2CCCC2O)C(=O)NC(C)C)cc(Br)cc2nc[nH]c12 C(C(O)CC(=O)NCC1CCOC1=O)NC(=O)COC1CC=CC1 CC(C)CC(C)(CNC(=O)C(C)c1ccsc1)NC(c1ccoc1Cl)=O c1(C(=O)NC2C(CC(=O)NCCCCCOC)CCCC2)cnccc1C#N CCC(O)C(C)C(=O)NCC1CN(C(=O)CC2CCCC3CC23)CCO1 N1(C(c2cnn(CCOC)c2)C(=O)NCC)CCC(C)(O)C1 N1(C(c2c(Cl)nc(OC)s2)=O)CC2ON=C(CNC(=O)C(=O)N(C)C)C2C1 C(=O)(C(CC(C)CC)NC(c1cnn(C)n1)=O)NCC(CC#C)(C)C c1(C(=O)NC(CCNC(CCC(=C)C)=O)C)cc(OC)ccc1F C(C(C)(C)CNC(c1ccc(F)o1)=O)N(C(=O)C(F)=C(C)C)CC c1(OC(C)C)ccc(C(N2CC(CNC(=O)CN(C)C)CC2(C)C)=O)c(Cl)c1 c1(C(N2CCC(CNC(C(C)Cn3ccnc3)=O)C2)=O)cc2cccc(Cl)c2o1 N1(C(c2ncn(CC)c2)=O)CC(F)(F)CC1C(N1CCOC(C)CC1)=O C1(C(=O)NCC(C(=O)OC)(C)O)CN(C(c2cncc(O)c2)=O)C2(CCC2)C1 c1(C(=O)OC)cc(C)cnc1N1CCC(NC(c2cnn(C)n2)=O)C(O)C1 c1(C2C(C(N3CCN(C(c4ccc(Cl)cc4)C)CC3)=O)C2)cccc(C#N)c1 C(=O)(C(C(=O)OCC)C(C)C)NC12C(CN(C(C=CCC)=O)C1)C2.OCC Cc1ccc([N+](=O)[O-])cc1C(=O)NCC1CCCN1CCN1CCCCC1C C1(NC(C2CCCN(C(c3c(OC(C)C)cccc3)=O)C2)=O)CCC2(CCC2)N1 CC1CC(c2nnnn2C2CCC2)(NCC2C(C)(C)C2(C)C)CO1 C(=O)(CN=c1cc[nH]cc1)NCC12C(CN(C(c3nc(OCC)oc3)=O)C1)CC2 C1(CC)CC(CC(=O)N(CC(C)(C)NC(=O)C=C(C)C2CC2)C)CCO1 CC(C)CCC(F)C(=O)NC1CC(O)C1CC(=O)NC12CCN(CC1)C2 c1(NCC2C(NC(Cc3c(C)ccs3)=O)CCCC2)ncc(S(C)(=O)=O)cc1Cl c1(CNC(Cn2nnc(=N)[nH]2)=O)ccc(CNC(=O)CC2CCC2)cc1F CN=c1nc(C(N2CC3CC(NC(c4cscc4SC)=O)CC2C3)=O)cc(C)[nH]1 C1(C(C)C)CNC(=O)CN1C(=O)Nc1ccnn1Cc1ccc(Br)s1 c1(-c2c(OC)cc(C(N3CC4CC4C3C#N)=O)cn2)cnc2n[nH]cc2c1 C(=O)(C(C)C(O)C(C)C)NC1CCN(Cc2cn(-c3ccc(C)nc3)nn2)C1 CCC(C(=O)NC1CCCC1NC(C1(C2CC2)CC=CC1)=O)C(F)(F)F N1(C(C2(C)CC2)=O)CC2CC(NC(=O)CC3CCCCC3(C)C)CC1C2 N1(C(CC2(OC)CCC2)=O)CCCC(NC(=O)CCc2nc(C)c(C)[nH]2)C1 C(=O)(CC(C)P(C)(C)=O)N1CC(CCCC)N(C(C2CCCC(=O)N2C)=O)CC1 C(CCCCCCCO)c1c(C)nc(-c2ccc(C)cc2O)s1 C12(C(N3C(C)(CNC(Cn4nc(C)oc4=O)=O)CCC3)=O)CCC(C1)OC2C S(=O)(=O)(c1cc(F)cc(F)c1)N1CC(F)CC(C(=O)Nc2cc(C)c(I)cc2)C1 Cc1ccc(C(N2CCC(NC(c3n[nH]cc3[N+](=O)[O-])=O)C(F)C2)=O)cc1F c1(C(=O)NC(CC)CNC(c2cc(Cl)ncc2O)=O)cc(C)cc2c1OCC2 N1(C(c2ccn(CC)c(=O)c2)=O)CCC2CN(C(C3CC(S(N)(=O)=O)C3)=O)CC12 O=C(NOCc1ccccn1)C(F)CC1CC(NC(=O)C(F)CC2CCOC2)C1 c1(CN2CCC(C(=O)NC3CCN(S(C)(=O)=O)CC3)C2)cc(O)cc2ccccc12 CC(CN=c1nc(O)c2c(ncn2C)[nH]1)NC(C1COC(C)(C)C1)=O CCCCCCC(=O)N1CC2(C1)CN(C(c1cc(C(C)(F)F)n[nH]1)=O)C2 CC(C)C(C(=O)NCCOC1CCN(C(=O)Cc2ccccc2Cl)C1)NC=O c1(C(=O)NCC(CC)C)cn(CCNC(=O)CC2CSC2)cn1 C(=O)(CS(=O)(=O)C1CC1)NC1CCCN(C(COC2(C)CCOCC2)=O)C1 N1(C(c2ccc(CC(C)C)s2)=O)CCCN(C(=O)CC2CCC(=O)NC2)C(C)C1 CC(C)CC(C(=O)NC(Cn1cccn1)C(=O)NCC(=O)N1CCCO1)N(C)C C1(NC(CC2C(C)CCN(C(c3nocc3Cl)=O)C2)=O)CCCC(C2CC2)C1 CC1(C)CCC2(CC1)CC2C(CC(C1CCCCC1)NC(=O)C=CC(F)(F)F)=O CCCC(C#N)C(=O)N1CCOCC(NC(c2ccc(CNC(C)=O)o2)=O)C1 c1(C(N2CCC(c3ccccc3)(C(=O)OC)C2)=O)cc(Cl)cnc1F c1(C(=O)NC(CNC(C(C)OCC(C)C)=O)CO)ccc2nc(Cl)nn2c1 C1(CNC(=O)CCCCCF)CC2COCC2N1C(c1ccc2sncc2c1)=O C1(C(N(C)Cc2ccc(C)cn2)=O)CC(O)CCN1C(=O)C(c1ccn(C)n1)C C1(CNC(C(CO)NC(C(C)C)=O)=O)N(C(=O)C=Cc2cscn2)CCC1(C)C c1(OC)ccc(CNC(=N)NCCC2CCCC(C)C2)c(O)c1 N1(C(c2cnc(NC(C)=O)o2)=O)CC=CC(NC(c2nsnc2O)=O)C1 C(=O)(C1=CCCOCC1)N1C(C=CC(=O)NC2CCN(C(CC)=O)C2)CCC1 c1(-c2cn3cnc(C(N(CC)Cc4ccccn4)=O)c3s2)cccc2c1CCC2 C(N=c1[nH]c2ccc(Br)cc2s1)C1(CCNC(c2cc(C)c(C)nc2O)=O)CC1 N(C(=NCCCF)NCC(N1CCCC1)=O)Cc1cc(C)cc(F)c1 C1(C(=O)NCC2CCCC2O)(OC)CCN(C(=O)CCC2CCOC2)C1 C1(C(N(CCC(C)C)CCCO)=O)COC(CNC(=O)C(O)C2CCC2)C1 N1(C(C=C(C)Cl)=O)CCCC(CN2CCN(C(c3c[nH]c(=O)cn3)=O)CC2)C1 CC1(C)CCC(C(=O)NCC=CCNC(c2ccc(-c3csnn3)cc2)=O)O1 c1(C(C(=O)NC2C(NC(COCC(=O)OC)=O)C2)(C)C)ccc2c(c1)OCCO2 c1(OCC(CNC)O)ccc(CN)c(C(F)(F)F)c1.c1(O)ccc(Cl)c(F)c1 CCCCC#CC(C)(C)NC(C1CC(NC(=O)C(CC)NC(C)=O)C1)=O Cc1ccc(F)c(OCC(=O)NC2CCCC2NC(=O)CCC2CCCO2)c1 C1(CNC(CSCCCC)=O)CCN(C(c2ccsc2Cl)=O)CC1O C(C1=NOC2CN(C(=O)C#CC3CC3)CC12)NC(C(C(C)C)CCc1ccccc1)=O Cn1cnc2nc(N3CCC4(CC3)CCC4(C)C)nc(NCC#CCCO)c12 C1(N(C)C(=O)NCC(c2ccccc2)C2CCC2)CC1(C)C1(C)CC1 c1(C(N2CC(OC)C(F)C2)C(=O)NCC2CC2)ccc(F)c(C(F)(F)F)c1 CCC(C)CC(C(=O)NCc1ccc(C)nc1O)NC(=O)CC1(C)CC1 N1(C(C(c2cccc(F)c2)C)=O)CC(NC(=O)Cc2ccn(C)c2)C(C(F)F)C1 c1(CC(=O)NCCCN(C(=O)C(C)(C)CCSC)CC)ccc([N+](=O)[O-])cc1F N1(C(CCCOCC=C)=O)CCC(C2CCN(C(c3cn(C)cc3C)=O)C2)C1 C(C(O)C(C)(C)CC(=O)O)NC(c1c(C)nc(-c2ccc(OCC)cc2)s1)=O c1(C(=O)NC2CN(C(C=CC)=O)C3(C2)CCOC3)[nH]c2ccc(OC)cc2c1C C(=O)(CCCC(F)(F)Br)NCCC(C)N(C(c1ccc(OC)nc1)=O)C N#Cc1cccc(CC(=O)OC2CCCN(C(C3(C(=O)OC)CC3)=O)C2=O)c1 C1(NC(c2ccc(NC=O)cc2)=O)CN(C(c2ccccc2)=O)CCC1CO C12(CNC(C3CCC(=O)N3C3CC3)=O)CCC(CC1)N(C(C1C=CCC1)=O)C2 c1(C(N(NC(=O)NC(C(C(=O)OC)NC(C)=O)C)C)=O)cc(=O)cc(Cl)[nH]1 C(C(=O)N=c1cc[nH]cc1Cl)c1nc(NC(c2scc(C)c2)=O)sc1 c1(N(C(CNC(C(C)CN2CCOCC2)=O)C)C)ncncc1Br Cc1ccc2c(C(=O)NC(CNC(C3CCOC3C)=O)C(C)(C)C)c[nH]c2c1 c1(C(N2CC=CC(NC(C3C(OCC)C3)=O)C2)=O)cnn2ccc(C)cc12 c1(CN2C(C(N3CCC(OC)C3)=O)COCC2)cc(Br)ccc1[N+](=O)[O-] C1(CN(C(=O)Cc2cccc(F)c2)C)CCN(C(C2(C#N)CCOC2)=O)CC1 c1(CC)ncncc1C(N1CCC(CCNC(=O)CSc2n[nH]c(C)n2)C1)=O Cc1sc(COC(=O)C(C(C)C)NS(C)(=O)=O)c(C)c1C N1(Cc2c(OC)c(F)ccc2F)CCC2(CCCN2C(=O)C(C)(C)O)CC1 CC(C(=O)NCCCCC(=O)NC1CCCC(F)(F)C1)C(F)(F)F CC1(C)CC1(C#N)C(N1CCC(CC(=O)NCC2CCC2CO)C1)=O C1(O)(c2cn(CC3CC(C)(C)OC3)nn2)CCCN(C(=O)CC2(CO)CC2)CC1 Cn1ncc2c1CC(CCC(=O)NNC(=S)NCCCN1CCOCC1)CC2 C(=O)(CCCC(=O)Nc1nccs1)NC1CC(CNC(c2cc(OC)ns2)=O)C1 CC1CC2(CCN(C(c3nncs3)=O)CC2)CN1C(=O)CC(C)CC(C)(C)C Cc1cc(CC(=O)N(CC(O)CN(C)C(c2coc(Cl)c2)=O)C)ccc1CO C(=O)(C(F)(F)CCn1cccn1)N1CC(F)(CNC(C2CCC(=O)O2)=O)C1 c1(C(N2CCC3(NC(C=Cc4n(C)ncc4)=O)C(C2)C3)=O)cc(S(N)(=O)=O)co1 C=CCC(C(=O)NC1CCC1NC(C1CC1C(F)(F)F)=O)NC(=O)OC(C)(C)C Cc1sc2ncnc(N3CCC4CCC(SCCCNC(=O)N(C)C)C34)c2c1C N1(C(C=CCOC)=O)CC2CCOCC2(NC(=O)CCc2nncs2)C1 N1(C(CSCCOC)=O)CCN(C(c2ccc(C(C)(F)F)cn2)=O)C2CCCC12 Cc1cnn(C(C)C(=O)NC2CC(CCNC(=O)Cc3cncn3C3CC3)C2)c1 C#Cc1ccc(F)cc1C(=O)NC1CCN(C(=O)C(F)C(=O)OCC)CC1(C)C N1(C(c2cc(SC)c(F)cc2)=O)CC2OCCN(C(=O)CSC3CC3)C2C1 c1(CCC(=O)N(CC(CC)NC(=O)C(O)C2CCC2)C)ccc(OC)cc1OC C1(C(N(CCC(=O)NCC2CCC(CO)CC2)C2CC2)=O)CC2(CCCO2)C1 C1(OC)CC(NC(c2cnc[nH]2)=O)C12CCN(C(c1cccc(C#N)c1)=O)CC2 C(=O)(C(CC(C)(C)C)OC)NC(CC)CN(C(=O)CCOC)CC N1(C(C=C(C)C(C)C)=O)CC2CCC1C(N=c1nnn(C)[nH]1)C2 C1(O)(C(CC)C(=O)NCCN(C(=O)Cc2ccsc2)C(C)C)CCCCC1 C(=O)(CCC(=O)NCCC1CC(NC(C2(C(F)(F)F)CCO2)=O)C1)NCCC C12(OC)CCC(C(=O)NC3CCN(C(c4cc(C)nn4C4CC4)=O)CC3)(CC1)C2 C1(C(=O)NC2C(CNC(C(CC)(C)C)=O)CCCC2)CC2(CCC2O)C1 n1(C(C(=O)OC)C)nnnc1CNCC(C)COc1ccccc1 C1(C(=O)NCC(C(C)C)NC(C(C)(C)NC(=O)NCCC)=O)CCCOC1C c1(OC)ccc2[nH]c(=NCCN3CCCC(C)C3)[nH]c(=NCC(N)=O)c2c1 c12cc(cs1)COCC(C)NC2=O.C(=O)(C=CC(=O)N(C)C)NC1CC1 N1(C(N)=O)CC(F)CC1C(N)=O.C1CS(=O)(=O)C1 C12(CNC(=O)CN3CCCC3)CN(C(c3nocc3C3CC3)=O)CC1CCO2 C1(CCO)(CC)CN(C(=O)C(C)NC(C2CCC(=O)N2)=O)C1 C1(O)(NC(COCCNC(C(C)SC(C)C)=O)=O)CC(CO)C1.C(C)(C)C C(C(C)C)(C(O)C(=O)N(CCCNC(c1ccn(CC(C)C)n1)=O)CCO)OC C1(C)(OCC#C)CCN(C(=O)CNC(=O)CCCC(C)C)CC1 c1(CC(N2CC(C#N)N(C(c3ccns3)=O)CC2)=O)ccc2ncccc2c1 c1(C(=O)OC)cncc(NC(=O)N(C2CCN(C)C2)C)c1C c1(C(=O)NC2C(NC(c3nc(CC)oc3C)=O)COC2)ccc2nc(O)sc2c1 Cc1c(CC(=O)NC(C2CC2C(=O)NCC23CC2C3)C)cnn1C CCC(C)CCCC(=O)N1CC(NC(c2ccc(F)cc2C)=O)C(O)C1 N1(C(CCCC2C(C)C2)=O)CCCC(CC(=O)NC23CCCC2OCC3)CC1 Cc1ccccc1C1CCCCN1C(c1cc(C(F)(F)F)n(C)n1)=O Cn1cnc2nc(N3CC4CCC(C3)O4)nc(NCCCOC3CCC3)c12 N1(C(c2c(CC)ccc(F)c2)=O)CC(C2CN(C(=O)C(F)CC)C2)C1 C(=O)(C#CC(C)(C)C)NCCCCN(C(c1n(C=C)nnc1)=O)C N#Cc1ccc(CNC(=O)C(N)Cc2ccccc2Br)cc1 c1(C(=O)NC(CC)CN(C)C(c2ccc(C)s2)=O)ccc2c(c1)COCCN2 C1(NC(CC(CCC)C)=O)CN(C(c2cc([N+](=O)[O-])nn2C)=O)CC12CCC2 Cn1cnc2cccc(C(=O)NC3CCN(C(=O)Cc4cn[nH]c4)C34CC4)c12 C1(NC(C2N(C(C)C)C(=O)COC2)=O)CCCN(C(C2(C)CCOC2)=O)CCC1 c1(C(N2CCC(NC(CC(C)C)=O)(CF)C2)=O)cc2scc(Br)c2[nH]1 C1(NCc2cncc(OCC)c2)CC2(C1)CC(NC(C1CCCCO1)=O)C2 C1(C(=O)NCCCC(C)NC(c2ccco2)=O)CNC(=O)C(C)(C)C1 C1(NC(c2cccc(CC)n2)=O)CN(C(c2cc[nH]c2C)=O)Cc2ccnn2C1 C1(NC(CCC(=C)C)=O)CC2CN(C(C3CCC(C(=O)OCC)CC3)=O)CC2C1 Cc1ccnnc1C(=O)NCC1(C(=O)N(C)CC2CCC(C)CC2)CCCC1 c1(C(N2CC(=C(CNC(Cc3n(C)c(S)nn3)=O)F)C2)=O)cc2n(n1)CCOC2 C1(NC(=O)CCC2CC2)CCC(O)CN(C(=O)C(c2cc(Cl)ccc2Cl)(F)F)C1 N1(CC(=O)NCC2CCC(NC(CC)=O)CC2)CCCc2sccc2C1=O c1(C(=O)NC2C3CC(O)C2N(C(=O)Cc2ccsc2)C3)cc2cc(Cl)ccc2o1 C1(C(=O)NCC2(C)CCCN2C(C2C3CCC(F)(F)C23)=O)CC(=O)NC(=O)C1 C(=O)(C(CC(N)=O)NC(=O)C=C(C1CC1)C1CC1)N(CCCCC=C)C C#CCC(C)(C(=O)N1CC(C)CC(C)C1)NC(=O)C(F)CCCC N1(C(C2C(OCC)C2)=O)CCC(O)(CCNC(c2cc(Cl)ccc2N)=O)CC1 C(=O)(CCN=c1[nH]c(C)cc(=NC2CC3CCCCCC3C2)[nH]1)NC CCC(CC)C(=O)NCC(c1ccccc1)NC(c1conc1C1CCCO1)=O c1(C(N2C(CNC(c3n[nH]cc3F)=O)CC2)=O)ccnc(Nc2ccccc2F)c1 C#Cc1ccc(C(=O)NC2CN(C(c3ccc(CC)[nH]3)=O)CC2C2CC2)c(C)c1 C(=O)(C1=CC2CCCC12)N1CCCC(NC(C2C(OC)CCCC2)=O)CC1 N1(CC(=O)NC(=O)C(c2ccco2)SC2CC2)CCC2(CCOC2=O)C1 c1(C(C)C(=O)NCCCCn2cc(C3CCCCO3)nn2)ccc(F)cc1 C(=O)(C(CC(C)C)C(N)=O)N1CCC(C(N=c2nc(C(=O)OC)[nH]s2)C)CC1 C1(NC(C2CC(C)C2)=O)CCN(C(=O)C(C)(C)CCC#N)CC12CCC2 N1(C(C2CCCC2CF)=O)CCCC(N(C(c2csc(F)c2)=O)CC2CC2)C1 C#CCC(C(=O)NC(C)Cc1cnc[nH]1)NC(=O)CCOC1COC1 N1(C(CC(=O)OC)=O)CCC(COC(c2ccc3nonc3c2)=O)OCC1=O C1(C(=O)NCC(CNC(C2CC3(CC(=C)C3)C2)=O)O)CCc2nc(CC)cn2C1 C1(NC(C(C)N(C)C)=O)COC2CN(C(=O)Cc3cccc(Br)c3F)CC12 C(=O)(C(C)(O)CCC)N1CC(C2OCCN(C(Cc3ccc(CC)cc3)=O)C2)C1 c1(C(=O)NC(C)CCCNC(=O)C=C2CCN(C)C2)cc(C(C)C)n(C(C)(C)C)n1 C(=O)(C(C)OC)NC(COC)COCCOCCOC(C)C c1(C(N2CCC(CNC(C(C)OCC)=O)C23CC3)=O)cc(F)cc(C)c1C CC1CCCN(C(=O)C(=O)NC2(CCNC(=O)CC3CCOC3)CCC2)C1 C1(c2nn[nH]n2)(C(N(C2CCCC2O)CC)=O)CCCC1 c12ccccc1NC2C.c1(COCC)cc(CC(C)C)on1 c1(C(N2CC3CCN(c4ncc(C5CC5)cn4)CC3C2)=O)cc2cc[nH]c2cc1Cl c1(OC)ccc2cc(NNC(=O)C3(C)CCN3)ccc2c1 CC1=NOC(=O)C1CC(=O)NC1CC(n2cncn2)C1 c1(CCCN2CC3C(C(=O)NCc4cnn[nH]4)C3C2)ccc(Cl)c(Cl)c1 N1(CC2(C)C(C)CNC2)CCc2c(cccc2[N+](=O)[O-])C1.N12CCC(C1)CC2=O C1(CNC(C2(COC)CCC2)=O)CC2(CCC2)CN1C(c1ncc(C)cc1C)=O CC(C)C(C)C(CNC(=O)CCCn1cccn1)NC(=O)CN(CC(C)(C)C)C c1(C(=O)NCC2C(C)CCN(C(CC(CC)O)=O)C2)ccc(C)c2c1CCCN2 Cc1ccc(C)c(C(N2CCOC(CN(C)C(C3CCOC3C3CC3)=O)C2)=O)c1 N1(C(C2C(C)CCC2)=O)C2CCC1CC(N(C(=O)C(O)C1CC1)C)C2 Cc1cc(C(=O)NC(C)(C)CCCNC(=O)CCC(C)c2ccccc2)[nH]c1C C1(N(C(C2CCCN(c3c(C)ncc(C)n3)C2)=O)C)CCC2(CCCC2)CC1 N1(C(C2(NC(C)=O)CCC2)=O)CCCC(C)(NC(=O)CC2CC2(C)C)C1 c1(C(=O)NC(C2(C(=O)NC3(C=C)CCOCC3)CC2)C)cccc2ccnn12 C1(NC(c2n[nH]cc2Br)=O)CCCC1CNC(C1CCCOC1)=O c1(CCC)cc(C(N2CCC(NC(=O)C(C3CCOCC3)OC)C2)=O)ccn1 C1(O)(CC#C)CCN(C(=O)CC(CNC(=O)C(C)(C#N)CC)OC)CC1 C(=O)(C(CCSC)NC(C1COCC(C)O1)=O)N(C(CSC)C)C c1(CC)ccc(F)cc1C(N1CC(O)(C(C)NC(C2CC2C(C)O)=O)C1)=O C1(NC(CC(C)=C(C)C)=O)C(CNC(=O)CS(C)(=O)=O)CCC12CCC2 N1(C(c2nnc(C)s2)=O)CCCCC1C(C)NC(=O)C=CCN1CCCC1 C(=O)(C(C)(C)C(=O)NC1CC2(NC(=O)C(C)N(CC)CC)COC1C2)OCC O=C(Nn1cccn1)C1CCN(C(c2ccccn2)=O)CCO1 c1(OC)ccc(C(=O)OCCOCCc2ccc(C)cc2)nc1 C(=O)(CC(O)C(C)(C)C)NCC1OCCN(C(C2(C(C)(C)OC)CC2)=O)C1 C(N=c1[nH]c(C(C)(F)F)cs1)C1N(CC(CCCC)O)CCCC1 C(=O)(C(C)(C)C1=CCSCC1)N1CC(CC(C)NC(c2ncn(C(C)C)c2)=O)C1 c1(CC)nc(C(C)NC(=O)C(C)N(C)C(c2ccco2)=O)no1 C(C(CCC)OC)NC(CN(C(=O)C(C)n1cccn1)CC#C)=O c1(OC)ccc2c(C(=O)NCC(C)NC(C3(CCF)CCC3)=O)cnn2c1 CC1CCCN(C(c2cc(C(C)(C)C)on2)=O)C1CNC(=O)CCC(N)=O CC1Oc2ccccc2OC1C(=O)NC1CCCN(c2nncs2)C1 C(C1=NOC2CN(C(=O)CCc3cncn3C)CC12)NC(Cn1c(C)ccn1)=O c1(OC)ccc(CN(CCN)CCc2ccccc2)cc1F c1(C(N(CCN(C(c2cscc2C)=O)CC)CC)=O)cc(O)c2c(cnn2C)c1 C1(C(C)NC(C2C(CC)C2)=O)CCN(C(C2(F)CCOC2)=O)C1 CC(C)CC(=O)N1CCC(C(=O)NCC2CCC(C)C2)O1 N1(C(=O)OC(C)(C)C)CCCC2CN(CCc3ccc(Cl)cc3Cl)CCCC12 C1(OC)CC(NC(=O)CC2CC3C=CC2CC3)CN(C(c2cc(O)ccc2Cl)=O)C1 c1(CNC(CC2C(C)CN(C(=O)CCCC3CCCO3)C2)=O)cccc(C#N)c1 C(C)(CS(=O)(=O)NC(c1ccc(Oc2ccc(Cl)cc2)cc1)=O)OC C(=O)(C1=CS(=O)CCC1)NC1C(NC(CCCCCOCC)=O)CCCC1 O=C(CCN=c1[nH]c(=NCC2CCSC2)[nH]c2cccnc12)NCCCCO N1(C(C(N2CCOC2=O)C)=O)CCCC(CN2CCC(N3CCCCC3)C2)C1 Cc1ccc(Cc2nc(-c3ccoc3)nn2C2CCC(C)C2)cc1Br Cn1c(-c2nc(Cc3cccc(F)n3)no2)ccc1C#N N1(CC)CCN(CCC(=O)NC2CN(C(=O)C=CC(C)(C)C)CC2C)CC1 CC(C)CC(CCc1ccccc1)C(=O)NCCC1CN(C(C2CC(C)C2)=O)C1 N1(C(CC(CNC(c2ccc(CC)o2)=O)OC)=O)CCOC2COCC12 Nc1ccc(Cl)c(C(=O)NC2CC2CNC(c2ccnnc2S)=O)c1 N1(C(C2CC(C(C)C)C2)=O)CCN(C(c2ccc([N+](=O)[O-])o2)=O)CC1C1CC1 CCCCCCCC(F)C(=O)N1CCC(NC(=O)CSCC(F)(F)F)C1 C(=O)(CCC(=O)NCC1(C)CCN(C(=O)CCC2(C)CC2(F)F)C1)OC c1(N(CC=C)C)ccc(C(F)(F)F)cc1S(=O)(=O)N1CCSCC1c1nccs1 c1(CCC)onc(C)c1C(=O)NCC1(F)CC(NC(c2[nH]c(C)nc2C)=O)C1 c1(NC2CCC(SCC)CC2)ncnc(N(C)Cc2nccn2C(F)F)c1C CCCN=C(NC1CNC1)NC1CCN(c2ccccn2)C1.C1C2(CC2)C12CC2 c1(C(=O)NCC2(CNC(C(F)=CCC)=O)CC2)ccccc1OC C1(N(C(=O)CCOCCCNC(=O)Cc2cnns2)CC=CC)CCN(C)CC1 C1(CNC(CC2CC(=C)C2)=O)CCC2(CN(C(c3cncc(Cl)c3)=O)C2)O1 Cc1cc(NC(=O)C(CO)NC(=O)C=Cc2ccncn2)cc(C#N)c1 Cc1ccc(-c2ccc(C(C)NC(c3ccncc3)=O)cc2)c(C#N)c1 c1(C(C(=O)NC2(C)CCN(C(=O)OC(C)(C)C)C2)=O)c[nH]c2ccccc12 C1(CNC(C=C(C)C)=O)CCN(C(C2CC3(CSC3)C2)=O)C12CC2 N(C1c2ccccc2CCCC1C)NC(c1c(CC)onc1C)c1nnnn1CC c1(C(=O)NCCC(CCNC(C(CCC)C#N)=O)C)ccc2cc(F)ccc2n1 c1(C(C)C)ccc(C(=O)NC(C)CN(C)C(C2(C(N)=O)CCC2)=O)c(O)c1 N1(C(c2c(C)cn(C)n2)=O)CC2OCCN(C(C3CCC3n3ccnc3)=O)C2C1 C1(C)(C(=O)OC)CCN(C(=O)NC(c2ccncc2)C(C)C)C1 C1(CNC(c2c(C)[nH]c(C)c2C)=O)CN(C(C2(CC)CCCO2)=O)CC(C)(C)O1 N1(CC)CCCC1CN(C)C(c1csc(CNC(=O)C(F)n2ccnc2)c1)=O N1(C(C(c2[nH]c(=N)sc2)(F)F)=O)CCCCC(CNC(=O)CCc2cnco2)C1 c1(C(N2CC(CNC(C=C(C)c3cccs3)=O)C(C)C2)=O)c[nH]c2nccc-2c1 CCC(CC(=O)NC1CC2(C1)CC2NC(=O)Cc1ccc(C(C)=O)s1)C(C)(C)C C(=O)(C(C)(C)CCSC)NC1CC(OCC(=O)NC2CC(C)(CC)C2)C1 C1(CNC(C=CC2N(C(CC(CC)SC)=O)CCC2)=O)OC(=O)CC1(C)C N1(CC(C)NC(CC(C)F)=O)CCN(C(=O)CCCn2cccn2)CC1 C1(C(c2nnnn2CC2CC2)NC(c2cscn2)C)CCCC1(C)C N1(C(C2(CCOC)CCC2)=O)CCC2(CCN(C(=O)Cc3ccc(C)s3)C2)C1 C1(CNC(c2cnn(C)n2)=O)CCCCN(C(C2CCCNS2(=O)=O)=O)C1 Cc1nnc2n1CCC2(C)C(=O)N1CCC1CNC(c1cncc(N(C)C)c1)=O c1(OCNc2c(-c3cc4c(cc3)NC(=O)NC4)csc2)ncc(S(=O)(=O)O)cc1Br CC1CCCC1(C(=O)N(C)CCC1CCCO1)NC(c1cnn(C)n1)=O N1(C(c2c(C(C)C)ncs2)=O)CC2C(CNC(=O)C(F)=CC3CC3)C2C1 C(C(C)(O)CNC(=O)C(C)c1ccco1)NC(C1(CC(C)C)CC1)=O CC1CCC(C(=O)Nc2ccnc3[nH]cnc23)CC1(C)C N1(C(COC)=O)CCC(C2CCN(C(=O)CC34CCC(CC3)CC4)CC2)CC1 CCC(C)(CNC(c1cc(C#N)n(C)n1)=O)C(=O)Nc1cncc(F)c1 C1(NC(C(CCC=C)(C)C)=O)CC2CCC(C1C)N2C(=O)OC(C)(C)C c1(C(N2CC3CN(C(C(C)Sc4ccccn4)=O)CC32)=O)cc(F)c(Cl)cc1F c1(C(=O)NC(CNC(c2ccc(CC)o2)=O)C)csc([N+](=O)[O-])c1 C(=O)(C1=NN(C)C(=O)CC1)NCC1C2N(C(C3(COC)CC3)=O)C(CC2)C1 N1(C(C(C)N(CC)CC)=O)CC(C(=O)NCCC(=O)N(C)C)C2(CCC2)C1 C1(O)(C(C)Nc2nccnc2F)CCN(C(=O)CCc2ccc(F)cc2)CC1 CC(C)C(O)CC(=O)NC(C)(C)CCC1CCN(C(=O)C2=NOCC2)CC1 CN1CCC(C(=O)N(CC(O)C2CCC2)C)(NC(C2CC2[N+](=O)[O-])=O)C1 C1(C(=O)NCc2ccc(SC)cc2)CC2CCC1N(C(c1cc(O)n(C)n1)=O)C2 C(=O)(C#CC1(C)CCCO1)N1C(=O)C2C3CC(CC23)C1.C12(CC)CCC(N=[N+]=[N-])C1C2 CCC(C)(C(=O)NC(CNC(C1(C)CCSCC1)=O)CO)OC N1(C(c2ccc(S(C)(=O)=O)o2)C(=O)NCC2CCOC2)CC2CS(=O)(=O)CC2C1 C1(NC(C2CCC(CC)O2)=O)CN(C(c2ccoc2C(C)C)=O)CCC12CCC2 N1(C(c2ncc(I)s2)C(=O)NCC=C)CCOc2cc(Cl)ccc2C1 CCC(CC)(CC)C(=O)N1CCC(C)C(NC(c2cc(CCCO)on2)=O)C1 C(=O)(C1=Cc2ccccc2OC1)N1C(CNC(c2c(CC)nco2)=O)COCC1 S(=O)(=O)(c1sccc1C)NC(CC)(C)C(N)=O N1(C(C(C)(C)O)=O)CC(NC(c2ccc(-c3ccncc3)o2)=O)CC(F)C1 CC(C)(CC1CCOC1)C(=O)NCCC1CCN(C(C2CCCC(=O)N2)=O)CC1 c1(C(N2C(CN(C(=O)C(F)C3CC3)C)CCC2)=O)ccncc1F C1(C(=O)NC2C(NC(CNC(CCC)=O)=O)CCC2)Cc2ccc(C)cc2S1 CC1=NOC(C)(C(=O)NCC2(NC(c3c[nH]nc3Br)=O)CCOCC2)C1 N1(CC2CCCC(CC)C2)CC(=O)N(CCc2cnc(C)o2)C1=O C1(CC(=O)NCCN2CC(OC)C2)CCC(NC(c2[nH]ccc2C(=O)OC)=O)C1 C(C(=O)N=c1ccn(C(C)CC)[nH]1)C1(NC(C(CCC)C#N)=O)CCCC1 N1(C(C(C)Cn2ccnc2)=O)CCC(O)(CNC(=O)CC#N)CC1 C1(NC(C(CC)N(C)C)=O)CCN(C(c2ccc(C#N)cc2O)=O)C12CCCC2 CCCCCC(O)C(=O)N1CCC(CNC(c2cc3ccsc3n2C)=O)C1 C1(NC(C(C)(O)C2CCC2)=O)CN(C(=O)C(CO)NC(N)=O)Cc2nccn2C1 C1(C(C)(C)NC(C=CCOC)=O)CCCN1C(c1cc(Cl)c[nH]1)=O c1(C(N2CCC(C(=O)NC3C=C(C)CCC3)(CO)C2)=O)cc(O)ccc1F CCCC(CCC)C(=O)N(CC(C)C(N1CC(CO)CC(C)(C)C1)=O)C N1(C(C(C)NC(c2c(C)onc2)=O)=O)CCOC(CN(C(=O)C(C)(C)O)C)C1 C#CC1(CNCC(c2ccn(C3CC3)n2)C2CCCS2)CCC1 c1(C(=O)NC2CN(C(COCC=C)=O)CC2O)ccc(N)c(OC)c1 C=C(C)c1ccccc1NC(=O)CCC(C)NC(=O)CCc1ccco1 N1(C(CCSCC)=O)CC(C2CCN(C(c3ccc4c[nH]nc4c3)=O)CC2)C1 C#Cc1cnc(NC(=O)C(CCC2CCC2)NC(=O)C(C)OCCOC)c(C)c1 c1(C(N(C2CCN(C(CC(C=C)(C)O)=O)C2)C)=O)ccc2c(c1)CC(C)(C)O2 c1(COC)ccc(F)cc1NC(=O)CCc1cccc(F)c1OC O=C1CCC(C(=O)NCC2(NC(=O)C=CC3CCOC3)CC2)N1 C(=O)(C(C)(C)C(C)NC(=O)CCOC(C)=O)N1CCC(OC)C1 C=CC(O)(C(=O)NC(C)CN(C(=O)Cn1cnnc1O)CC)C(F)(F)F c1(C(C)C)nc(NCC23CCCC2C3)cc(=NC2CCOC2c2ccnn2C)[nH]1 C1(C(=O)OCC)CC12CCN(C(=O)Oc1cncc(F)c1)C2 C1(C(=O)Nc2nc(Cl)cs2)CN(C(=O)CC=C(Cl)Cl)CC1c1ccccc1 C1(CNC(c2cccc(C3CC3)n2)=O)CC2CCC1N2C(c1ccccn1)=O c1(CC(=O)N(CCCNC(C2(F)CCOC2)=O)CCO)ccc2c(c1)CCOC2 N1(C(c2nn(C)c(O)c2)=O)CC2CCC2(CCNC(c2cccc(=O)n2O)=O)C1 N1(CC(=O)Nc2ccc(C(C(C)C)=O)cc2)CC2CC(C1)CS(=O)(=O)C2 c1(C(N2CC3(CN(C(C4(C#N)CC5CC5C4)=O)C3)C2)=O)nc2c(s1)COCC2 c1(C(N(CC(CN(C(c2ccc(CCC)cc2)=O)C)O)C)=O)ccnc(Cl)c1F C(=O)(C(CCC1CCC1)N1CCSCC1c1ccccc1)N(C)C1CC1 c1(C(N(CC(CNC(C(C)OCC=C)=O)C)C)=O)cnn(C2CC2)c1 N1(C(C(SC)SC)=O)CCC(C)(NC(CSCC(N2CCOCC2)=O)=O)C1 N#Cc1cccc(O)c1NC(C1CCC(Nc2cc(C#N)ncn2)CC1)=O c1(C(=O)NC(CN(C(C(C2CC2)SC)=O)C)C)[nH]cc2c1CCCC2 Nc1ccc(N2CCCC2)c(C(=O)NCC2CCCC(F)(F)C2)c1 c1(NC(c2cccs2)=O)cccc([N+](=O)[O-])c1.c12csc(c1)C(=O)NCC(=O)N2 CCCCC(C)(F)C(=O)NCC(C)(C)CN(C)C(C1CCOC1(C)C)=O C(C(O)CO)N(C(=O)C(=O)N(CC(C)C)C)CC N1(C(C2(C=C)CCOCC2)=O)CC2CCC(NC(C3(C(C)C)COC3)=O)CC2C1 C1(C2CCC2)(C(N(C2CCN(C(C3COC(C)(C)C3)=O)C2)CC)=O)CC1 C1(C(=O)NC2CC(CNC(C=CCN(CC)CC)=O)C2)CCC(CSC)CC1 N1(C(N)=O)CCCN(C(c2ccccc2Cl)=O)CC1.C(C(=O)OC)N(CC(=O)NC=O)C N1(C(C2CC(OC)C2)=O)CCCC2C1CCCN2C(c1ccc(C)o1)=O c1(NC(N(C(C)C)CCN(C)C)=O)ccc(OC(F)F)cc1F C1(C2CC2)(C(N(CC)CC2CCN(C(c3coc(O)n3)=O)CC2)=O)CCOCC1 Cc1ccc(C#N)cc1NC(=O)CC1C=CC(NC(c2cccn2C2CC2)=O)C1 N1(C(C(COC)N(C)C)=O)CCC(N(C)C(c2ccc(N(C)C)nc2)=O)CC1 C(=O)(C(C)(C)C(F)(F)F)N1CC(CNC(c2ccc(CC)s2)=O)OCC1 CC1CCN(C(C2C=CCC2)=O)CC1CNC(c1cc(C2(Cl)CC2)n(C)n1)=O C(C(=O)N1CC(N(C)C(C2CC3(CSC3)C2)=O)C1)(C(C)(C)C)c1ccc(C)cc1 c1(CC)noc(C(=O)NCC2(F)CC(CNC(C3(C)CCOC3)=O)C2)c1C n1(CC)nccc1C(=O)NC(C1(O)CN(C(=O)C(N2CCNC2=O)C)C1)C CS(=O)c1ccccc1-c1cn(C2CC3(C2)C(CO)C3(F)F)nn1 c1(CC)cccc(F)c1C(=O)NCCOCCCNC(=O)C(C)Cn1ccnc1 c1(NC(C2CN(c3c(OC)ccc(OC)c3)C(=O)C2)=O)ccc2c(c1)C(=O)CC2 c1(C(N2C(C(C)NC(C3CCCCC3O)=O)CCC2)=O)cc(O)nc(N(C)C)n1 N1(C(C(c2ccccc2)OCC)=O)CCN(Cc2cccc(OC)c2)C(=O)C1C c1(CC)occ(C)c1C(N1CCC(n2cc(C3CCCC(=O)C3)nn2)C1)=O c1(CC(=O)OC2CC(=O)OC2)cc(F)c(F)cc1O C1(CNC(C2CC2(F)F)=O)CC(C(=O)N(C2CCOC2)CCO)=NO1 N1(C(C=CC=CCC)=O)CCC(NC(c2cn(C)c(C(F)F)n2)=O)C(C)(C)C1 c1(NC(=O)C(N2CCCC2CC2CCCCC2)=O)nc2ccsc2s1 c1(CC)cc(C(=O)NCC2CC(C)(C)CN2C(c2ccnn2CC)=O)c(C)nn1 CN1CCN(C)C(C(N2CCN(C)C(C(=O)N(C3CCSC3)C)C2)=O)C1 c1(C(=O)OC)cc2c(NC(c3cc(C)ccn3)=O)cccc2s1 c1(C(N(CCNC(=O)Cc2ccc(O)cc2Cl)CC)=O)ccc2nnnn2c1 N1(C(C2(C=C)CCC2)=O)CCOC(C2CN(C(C3CC=CCC3C)=O)C2)C1 CC(CNC(c1csc2c1CCCC2)=O)N=c1nc[nH]cc1C#N c1(-c2c(COC(C)=O)cccc2)c(CCO)nn2c1CCCC2 C1(C(N(CC#C)CC2CCCO2)=O)CCCN(C(c2cccc(NC)n2)=O)C1 CC1(C(=O)NCC2C3CN(C(c4cocn4)=O)CC23)CCCCC1(F)F C=CCC(C)(C)CC(=O)N1CC2CC(NC(c3snc(O)c3Cl)=O)C1C2 N1(C(CCC2(C)CN(C(c3cc(C(C)=O)[nH]n3)=O)C2)=O)CC2(CSC2)C1 N1(C(C=CCOC(C)(C)C)=O)CCc2nc(CNC(=O)CCC(C)(C)F)sc2C1 C(CN=C(NCC(F)F)NCC1CC(F)C1)OC C1(NC(C(C)CO)=O)CCC2(CC1)CCN(C(=O)C#CC1(C)CCCCO1)C2 c1(OCC(=O)N(C)CC2CCN(C(C(CC)OC)=O)CC2)ccc(C)cc1F c1(C(N2CC(CCNC(C3CCC4CC4CC3)=O)OCC2)=O)n[nH]c2c1CCC2 Cc1ccc2c(cnn2C)c1-c1cc(C(=O)Nc2cc(F)cc(F)c2Cl)n[nH]1 C(=O)(C(CC)OC)NCC(CC)NC(=O)Cc1nc(C)no1 C1(C(=O)NC(c2cn(CC)nc2)C)C(O)CCN1C(c1cnsc1)=O S(=O)(=O)(c1cc(F)cc(Br)c1)N1CCCC(C)(C(=O)NC)C1 c1(C(N2CCC(NC(C3(Cl)C(C)(C)C3)=O)C2)=O)cccc(Cl)c1O C1(OC)CCC2(C(N3CCC(CNC(c4cnc(C(F)(F)F)s4)=O)C3)=O)CC12 C(C(O)CC(=O)N1OC2CCC1C2)NC(C(C)NC(CC)(C)C)=O C1(C(N(C2CCCC2)CCCNC(=O)CC2CCC2)=O)C2C3CCC(C3)C12 C12(C(N(C(C)CNC(=O)C(C)(C)c3ccnn3C)C)=O)CC1COC21CCC1 C#CCC(C)(CC)C(=O)N1CCN(CC(=O)NC2CC3(C2)CC(C#N)C3)CC1 CCCCCCCCCC(=O)NC1CC2CC(NC(C3(F)CC3C)=O)CC12 c1(C(=O)NC2C(NC(CCN(CCC)C)=O)C2)c[nH]c(Br)c1 Nc1ccc2c(c1)CCCN2C(c1ccc(C(F)(F)F)o1)=O c1(C(N2CCC(C(C)(C)C)(CNC(C(C)CF)=O)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C(CC(C)(C)CN=c1[nH]c(=NC2CCS(=O)C2)[nH]c2c1CCCC2)OC Cc1[nH]nc2ccc(C(=O)NC3C4CC3N(C(C3(COC(C)C)CC3)=O)C4)cc12 C1(C(=O)NC(C2CCN(C(c3c(C)nncc3)=O)C2)C)CC2CC1C1CC21 CC1(C)C(CC(N2CCC23CCCC3)=O)CCN1C(=O)C=CC1CCOC1 N1(C(Cc2cc(C)n(C)n2)=O)CC(NS(=O)(=O)c2cccnc2)CC(F)(F)C1 C(=O)(C(C)CC)NCC(=O)NCC(=O)N(CC(CC)O)C1CC1 Cc1nc2ccc(CNC(c3cnc4cc(C)ccn34)=O)cc2[nH]1 Cc1ccc(C)c(C(=O)N(C)C)c1.N12CC3CCC1C3C(=O)NOCC2=O c1(OC)ccc(C(=O)NC2CCCC(NC(=O)CNC(=O)C3CC3)C2)c(N)c1 c1(C(=O)NC(C2N(C(c3ccc(SC)o3)=O)CCC2)C)nc2cc(F)ccc2s1 c1(C(=O)NCC2CC(NC(CC3C(=O)NC(=N)S3)=O)C2)coc2cc(O)ccc12 CC(C)CC(C(=O)NCCC1(CCNC(C2(F)CC2)=O)CC1)N(C)C c1(OCC)cc(OCc2nnc(C(F)(F)F)s2)nc(S(C)(=O)=O)n1 c1(C(C)Nc2ccc(N3CCCCC3)c(C(=O)O)c2)ccc([N+](=O)[O-])cc1F c1(C(=O)NCCC(C)N(C)C(C2CCOC2)=O)ccc2oc(O)nc2c1 Cc1cc(Cl)ncc1CC(=O)N(C1CN(C(=O)CN2CSCC2=O)CC12CC2)C CC1(C)COC(CCC(=O)NCCC(O)CNC(=O)C=CC2CCC2)C1 c1(C(=O)NC2CCCC(C(=O)OCC)C2)c(C)[nH]c2c(OC)cccc12.C1CN1 C(=O)(C1c2c[nH]nc2CN1C(=O)Cc1cnoc1)NCCC1CCN(C)C1 C=Cn1ncc(C(=O)NCC2(C(=O)N(C(C)CO)C)CC3(CC3)C2)c1N N1(CCNC(C2(F)CCC2)=O)CCCN(C(C2(F)CCCOC2)=O)CC1 C(CCC(=O)NCCC1CCN(C(c2cc(C)co2)=O)C1)=CC C1(C(=O)OC)(C(=O)OC)CCC(NC(=O)N(c2ccc(Br)o2)C(C)C)C1 c1(C(N2CC(C(C)NC(Cc3cc(C)no3)=O)OCC2)=O)ccc2nccn2c1 N1(C(c2cccc(OCC(C)C)c2)=O)CCN(C(=O)CN(C)C2CC2)C(CO)C1 c1(OC)cc(Br)ccc1C(=O)NC(=O)C(C)OC(=O)CSC n1(Cc2n(C)nnc2)nc(-c2ccc(Cl)cc2)nc1C(N)=O c1(C(N2C(CNC(C3CC4(CCCCC4)C3)=O)C=CC2)=O)cn2cccnc2n1 C1(C(N2CCC(NC(c3ccc(C(F)F)c(Cl)c3)=O)C2)=O)(CC)CCC(O)CC1 C(CCCCN=[N+]=[N-])NC(CC(C)CNC(C1C2CCCOC12)=O)=O C12(OC(CNC(=O)Cc3ccno3)=O)CCC(CC1)C2 C1(C(=O)NCC2N(C(C3(CN(C)C)CC3)=O)CC2)CC(c2cccnc2)=NO1 S(=O)(=O)(c1ccc(C)c(C(N2C3CCC2CN(C(C2CC24CC4)=O)C3)=O)c1)NC C1(CNC(C2CSCCS2)=O)CCN(C(C23CCC(F)(CC2)C3)=O)C12CC2 N1(C(CC(CNC(=O)C=Cc2ccsc2)OC)=O)CCC(F)(F)CC1 C1(C(N2CC(C)N(CC)CC2C)C(=O)NCCC)C2(CCC2)C12CCC2 c1(C(=O)NCC2(C(N(C)CC3(C)CC3(F)F)=O)CC2)cnn2c1OCC2 C1(NC(C(CCC)O)=O)(COC)CCN(C(C2CCC(=O)N(C)C2)=O)CC1 C(CCC(C(=O)NC(C1(O)CCC1)C)NC(c1cnc(O)c(F)c1)=O)OC Cc1cc(Cl)c(C(=O)NC23CCC(CN(C(c4cnccn4)=O)C2)C3)cc1F c1(NC)ccccc1C(=O)NCC(C)NC(=O)C(CCSC)OC c1(CC)nc2ccc(Cl)cn2c1C(=O)N(CCCN(C)C(c1cocn1)=O)C C12(CCNC(Cc3c(C)noc3C)=O)CCC1CN(C(c1ncncc1Cl)=O)C2 C1(c2cccc(OC)c2)CN(C(=O)C=CSC)CCN1C(=O)CN1CCC(C)(C)C1 CCC(CC)CCCNC(=O)CC1(NC(=O)C(C#N)C(C)C)CC1 N1(C(C(CC(C)C)N(C)C)=O)CC(F)(F)CC1(C)CNC(=O)CCN1CCOCC1 c1(C(N(C(C)CNC(=O)CCCOC(C)C)CC)=O)cc(C(F)F)cs1 c1(C(=O)NC2C(CNC(CN(C(=O)OCC)C)=O)CC2)nccc2ncccc12 c1(C(=O)NC2(C)CC(NC(C(C3OCCC3(C)C)C)=O)C2)cc(F)c(O)c(Cl)c1 c1(C(C)C(=O)NC2CC(CCNC(C34CCC(C3)C4)=O)C2)cccc(F)c1 C(=O)(C1=COCC1)NCCOC(C)(C)CNC(C1C2CCCC12)=O c1(CC(=O)N(CCNC(C2C(CC)OCC2)=O)C2CC2)ccc2nn[nH]c2c1 c1(CN(CC=C)CCNC(=O)C(C)C2CC2)noc2c1CCCCC2 N1(C(c2c(SC)cccc2)=O)CCN(C(=O)CC2CCOC(C)(C)C2)C2CCC12 CC(C)CCC(O)C(=O)NC1CCC(NC(=O)Cn2ncccc2=O)CC1 c1(CC(=O)N(CCCNC(CCC(C)SC)=O)C)nc2ncccn2n1 N1(C(Cc2c(C)cco2)=O)CC(C)(C)CC1CNC(=O)CN(C)C c1(C(=O)NC2CCN(C(c3c(C)sc(Cl)n3)=O)CC2F)cnc2[nH]ccc2n1 c1(CCCC)ocnc1C(=O)N(C)CC1CCN(C(=O)CSc2nnnn2C)C1 N1(C(=O)NC(c2ccc(C(F)(F)F)o2)C)CC(CN(C)C)C(N)C1 CCCC(C(=O)NC1CCCCC1NC(=O)C(c1ccc(C)cc1)(C)O)N(C)C CC(C(=O)N(CCCN(C(=O)Cc1csc(NC=O)n1)C)C)S(N)(=O)=O c1(C(=O)NC2(CC=C)CCN(C(=O)CCC(C)OC)C2)nccc2cc[nH]c12 C1(NC(=O)OC(C)(C)C)CC2CCCC(C1)N2C(c1ccnc(F)c1O)=O c1(CC(C)N(C(=O)C(=O)N)C2CC2)cccc(F)c1F.N1(CC)CC=CCC1 CC(C)(CNC(C1CC(F)(F)CN1C(=O)CC1CC(=O)NC1=O)=O)C(F)(F)F N1(CCCOC)CCCC(N(C2CCCC2)C(=O)CN2CCS(=O)(=O)CC2)CC1 CN1CC=CCC1CC(=O)NCCCOC1CCN(C(c2c[nH]cc2Br)=O)CC1 c1(C(=O)NCc2scc(C(N(C)C)=O)n2)ccc(C(C)(C)C)cc1N C(=O)(CCCN(C)N=O)N(C)CC1CCCN(C(C2N(CC)CC2)=O)C1 CC1(C)CCN(C(=O)C2=CCCSC2)CC1NC(C1C=CCCC1)=O C1(NC(=O)COCCCF)CN(C(c2cncc(CO)c2)=O)CC12CCC2 C1(C(=O)NCCCNC(=O)C2=NOC3COCC23)CC2(CCC(F)(F)CC2)CO1 CC1CC1(C#N)CNC(=O)C=CC(=O)N(C1(c2cc[nH]n2)CC1)C c1(C(=O)NC(CCNC(C(CC)(CC)CO)=O)C)nc(C2CC2)n2ccccc12 CCC(COC)C(=O)N1CCC(C(=O)NCc2cc(C3CC3)no2)O1 C1(C(=O)NC(CC)C(C)(C)C)COCCN(Cc2ccc(Cl)cc2OC)C1 C1C2CN(C(c3nc(C(CCCOCCOCCOC)=O)no3)=O)CC12.OC c1(OC(C(=O)NCCN(C(CC(C=C)C)=O)C)C)ccc(F)cc1Cl C1(CCNC(C2CCC2(F)F)=O)CCN(C(c2nocc2Cl)=O)C1 N1(C(COCCCCC)=O)CC(C)C(NC(=O)CSc2ccccc2)C(C)C1 C12(CNC(Cc3c(CC)con3)=O)CCC(CN(C(=O)CCC(CC)OC)C1)C2 N1(C(c2ccc(CC)[nH]2)=O)C2CCC1C(F)C(NC(=O)CC1CCCCO1)C2 c1(-c2ccc(Cc3nc(C)nn3C3CCCS(=O)(=O)C3)cc2)cc2occc2n1C C(CC(C(=O)NC1CC(CO)C1)NC(=O)C(c1cnn(C)c1)C)OCC N1(C(Cc2n(C)ncc2Cl)=O)CCN(C(=O)COC2CC2)C(CCO)C1 c1(C(CN(C(C)C)C(c2csnc2Br)=O)O)ccccc1 C1(COC)CN(C(c2scnc2Cl)=O)CCN1C(=O)COc1cccnc1 CC1(F)COCCN(C(C2CCC(F)(F)CC2)C(=O)Nc2ccccc2)C1 c1(C(C)NC(=O)N(CC2CC2)CC2CC2)cccs1 N1(C(c2c(C)ccc(C(N)=O)c2)=O)CCC(C)(C)C(NC(=O)CCCC2CC2)C1 N1(C(CC=CC=C)=O)CC2CCCC2(CNC(=O)CSc2ccc(C)cc2)C1 c1(C(N2CC(CC(=O)Nc3ccc(C)cc3)(OC)C2)=O)ccc(CO)c(F)c1 N1(C(C(C)OCCC=C)=O)CCN(C(=O)CC2CCCS(=O)(=O)C2)CC(C)(F)C1 Cc1ccc(CCC(=O)NC2CN(C(=O)C(C)Cc3cnc[nH]3)CC2C)c(C)c1 c1(C(=O)NCC2CC(NC(c3cc(C4CC4)on3)=O)C2)ccc2oc(=O)oc2c1 N1(C(c2c(C)cc[nH]2)=O)CCN(C(c2c(C)nn(C)c2Br)=O)CC(C)(F)C1 c1(C(=O)NCCOC2CN(C(C(C)=C(CC)C)=O)C2)[nH]cc2c1CCCC2 c1(C(=O)NCC2N(C(CC(C=C)C)=O)CC(COC)C2)cc(C(C)C)nc(O)c1 C1(NC(C2C(C(=O)NC(C3(C)CC3)CO)C2)=O)CCOCC1 C(=O)(C(O)CCNC(=O)CCc1ccncn1)NCCC(C)N1CCCC1 Cc1ccc(NC(N2CCC(O)CC2C)=O)c(Cl)c1 N1(C(c2c(CC)n(CC)nc2)=O)CCC2(CCN(C(C3CCNC3=O)=O)C2)C1 c1(C(=O)NC2CCN(CCCOC)CC2C)ccc2nc(C)cn2c1 c1(C(=O)NCCOCCNC(CC2(C)CC2(F)Cl)=O)ccc(=N)[nH]n1 Cc1cccn2nc(C(=O)N(C)CCN(C(=O)Cc3sccc3Br)C)cc12 C(=O)(CCCC(=O)C(C)(C)C)N1CCC(N(C(C)C)CCO)CC1 C12(CNC(c3c(CC)noc3)=O)CCC1CCN2C(=O)C(C)=CC(C)(C)C c1(C(N2CC(NC(C(C)P(C)(C)=O)=O)CC2(C)C)=O)n[nH]c2c1COCC2 N1(C(Cc2cnc(C)[nH]2)=O)CCCC(N(C(=O)CC2(C#N)CCCCC2)C)CC1 Cc1nc(N(C)CCN(C)C(C2CC=CCC2C(F)(F)F)=O)c(F)c(C)n1 C1(C(=O)NCCCCC2CN(C(C3CCC(CC)O3)=O)C2)CCC(O)CC1 c1(N(CC)CC)ccc(C(N2CCC(CNC(=O)C(C)(O)C3CC3)C2)=O)c(O)c1 N(C1c2ccccc2CC1NC(C1CC(CC2CC2)C1)=O)C(=O)C1=CCCCO1 CC(C)C(CNC(C1CC2C=CC1O2)=O)C(=O)NCC(C)(CO)CO N1(C(COC)=O)CC(=O)NC2CN(C(C3CC(OC4CCN(C)C4)C3)=O)CCC12 C#CC(CNC(=O)C=CC(C)(C)NC(C1CCN(C)C1=O)=O)CC(C)(C)C N1(C(c2c(C)onc2)=O)CCC(NC(c2csc(Br)c2)=O)CC1C C12(NC(Cc3c(C)nc[nH]3)=O)CCCC1CN(C(c1cccc(O)c1F)=O)C2 N1(C(C23CC(NC(Cc4c(C)ccs4)=O)C(OC2)C3)=O)CC2CCN(C)CC2C1 c1(C(N(CCCNC(=O)Cn2ccnn2)CC)=O)csc2cccc(F)c12 c1(C(=O)NC2(CCCNC(c3c(C)nc(CO)s3)=O)CC2)nc(O)nc(O)c1N C1(NC(=O)CCc2ccon2)CCN(C(=O)CC2NC(=O)NC2=O)CC12CCC2 N1(C(CCc2n(C)ccn2)=O)CC(C)(C)CC1CNC(C1CC2(C1)CC21CC1)=O C1(SC)CCN(C(c2ccnn2COC)C(=O)NCc2ccccc2)C1 c1(C(C(=O)NC(CN(C(C=C(CC)C)=O)CC)C)C)cc(Cl)ccc1OC C1(N(C(CC2(NC(C)=O)CC2)=O)C)CN(C(=O)C(C2CC(F)(F)C2)O)CC12CC2 Cc1nc2ccc(C(=O)NC3CCCC3NC(=O)CCS(C)(=O)=O)cc2nc1C c1(NC(COCCCC)=O)ccc(NC(=O)C(C)Cc2cccc(F)c2)cc1C c1(CCC(=O)NCC(C(C)C)(C)NC(C2CCC(=O)O2)=O)nc2cccnc2[nH]1 C1(NC(c2n(C)nc3c2CCC3)=O)CCCC12CCN(C(c1ccsc1)=O)C2 N1(C(COC)=O)CC=C(C(=O)NC2CCCN(C3CC3)C2)CC1 N1(C(c2c(Br)cn(C)n2)=O)CCC(NC(=O)C=CC(C)(C)C)C12CC2 N1(C(c2cc(C)ncc2)C(=O)NCC2CCOC2)CCCC2(C1)N=N2 C(=O)(C(C)(C)C(F)F)NC(CC)CNC(C1(c2ccsc2)CC1)=O C1(NC(CN(C)C(=O)C2CC2)=O)CN(C(C2(C)CC2(F)F)=O)CC1(C)C N1(C(COC(CNC(c2ccc(CC)nc2)=O)(C)C)=O)CCC2OCCC2C1 c1(OCC(N2CCC(F)CC2)=O)ncc(CO)cc1Br CC(C(=O)N(CCC(C(C)(C)C)NC(C1(c2cccs2)CCC1)=O)C)C(F)(F)F c1(C(N2CC(NC(C3(C)N(C)CC(OC)C3)=O)C(C)C2)=O)cc(Cl)cc(F)c1N c1(OC)cccc(CC(=O)NCC2(OC)CCN(C(C3CC(=C4CC4)C3)=O)C2)c1 c1(CC(=O)NC2(C3N(C(CN(C4CCC4)C)=O)CCC3)CC2)sc(O)nc1O C1(C(N(C(CC)CC)CCO)=O)C(C)OCCN1C(C12C(=O)C3CC1C2C3)=O C(c1ccc2ncccc2c1)=CC(=O)NC1(C)CC(NC(C2CC3CC3C2)=O)C1 c1(C(C)C)nnc2n1CC(c1nc(Cc3ccccc3S(N)(=O)=O)no1)CC2 C(c1ccc(Cl)s1)=CC(N1C(CN(C)C(C2CCC(=O)N2)=O)CCC1)=O C1(CC#C)(NC(=O)Nc2ccccc2Cl)CCCCC1 C(=O)(CC(C(C)(C)C)NC(=O)C1=CC2C=CC1C2)N1CC(C)OC(C(N)=O)C1 C1(C(N2CCC3CN(C(c4c(C)c[nH]n4)=O)C3C2)=O)CC2(C)CCCN2S1(=O)=O c1(C(C(=O)NC2CC(N(C(c3cc(CC)c(C)s3)=O)C)C2)C)cccc(C#N)c1 S(=O)(=O)(c1ccc(NCC2(C(C)C)CCC2)cc1Cl)NCc1cccc(SC)c1 n1(CC#C)ccnc1Cc1nnnn1CCCF.CCCCCC c1(C(=O)NCC(CNC(C(CC=C)C)=O)(C)C)cscc1S(C)(=O)=O CN1CCC(CC(N2CCCC2CNC(=O)Cc2nn(C)cc2Cl)=O)CC1 C1(C(=O)NCC=CCC(=O)NC(c2onc(C)n2)C)CCC(C)(C)C1 C1(NC(C(C2CCC2)OCC)=O)CCCN(C(c2ccc(OC)nc2F)=O)CC1 C12(C(N(CC(CN(C(COCCN(C)C)=O)C)O)C)=O)CCCCC1C2 C(=O)(CCCCC(F)(F)F)N(CCNC(C(C)O)=O)Cc1ccccc1 CC1CN(C(=O)CSc2ccc(Cl)cc2)CC1NC(=O)C(C)CO C1(C2CC2)(C(=O)NCC(c2ccco2)OC)CN(C(=O)CC2CCOC2C)C1 C(C(C)(C)CN=c1[nH]c(C)cc(=NCCN2CCCC2=O)[nH]1)OC C=CC(O)C(=O)N(C1(C(=O)NCC(C)C#N)CCC1)C1CC1 CCCC1c2ccccc2CCN1N1CCC(NC(=O)C(C)C)C1 C(=O)(C1Cc2ccc(Cl)cc21)N1CC2CCN(C(c3c(C)ncnc3)=O)CC2C1 O=S(=O)(c1[nH]c(=NCCCC2CCOC2)ccc1Br)NC1CCn2ncnc2C1 c1(CC(=O)NC(C2N(C(c3c(C)cnnc3)=O)CCC2)C)ccc(Cl)nc1C C12(C(N(CCCOCC)C)=O)C(N(C)C)C3CC1C2C3.C1(CC(=O)N)CCCO1 C1(NC(=O)CSC(F)F)CCC(CNC(c2c[nH]nc2OCC(F)(F)F)=O)CC1 c1(NCC2OCCN(c3ccnc(SC)n3)C2)ccc2c(c1)CN(C)C2=O C1(C(=O)NC(C=C)C2(C(=O)NC3C(C(=O)OC(C)(C)C)C3)CC2)CC2(C1)CC21CC1 c1(CC)cc(NC(=O)C(C2CCC2)NC(=O)CC(CN(C)C)CC)cnc1C C(CO)(CN=C(NC1CCOCC1)NC1CCC(=O)NC1)OC C(=O)(C(C)CC(=O)NCCC1(O)CCN(C(C2CC3(CCCO3)C2)=O)CC1)OC C1(CNC(C2CN(C)C2)=O)CCCN1C(=O)Cc1nnn(C(C)(C)C)n1 C1(NC(c2c(C)nc(CCC)o2)=O)COCCN(C(=O)Cn2cnnc2)C1 CCCCC(C(=O)NCC1CC2(CCC2O)C1)NC(C1CC2C=CC1O2)=O c1(C(=O)NC(CNC(c2ccn(C(C)C)n2)=O)(C)C2CCC2)ccnc(CO)c1 C1(CCC)CCC(C(C(=O)NC2CCOC2)N(C)C(c2nccs2)C)CC1 C#CCCN=C(NCc1nn(CC2CC2)nc1C)NC(C1CC1)C1CC1 c1(CNC(N2CCOC(COc3c(C)cccc3)C2)=O)c(F)cc(I)cc1F C1(NC(Cn2c(C)ncc2)=O)CCC12CCN(C(=O)C(C)(C)C(N)=O)CC2 C1(NC(C(C=C)CC)=O)CN(C(c2c[nH]nc2Cl)=O)C2(CCCC2)C1 c1(C(CO)N(C(=O)C(Cc2csc(Cl)n2)NC(=O)OC)CC)ccc(Cl)c(Cl)c1 c1(SCC)cc(C(N2CC(CNC(c3csnc3OC)=O)C2)=O)ccn1 c1(C(=O)NC(CC)COCC2CC2)ccc(Br)s1 C1(n2c(-c3c(C)nc(C)[nH]3)nc(CCCCOC(C)(C)C)n2)CCC(C)(C)CO1 C12(CNC(CC3CN(C)C3)=O)CCCC1CCN2C(c1ccc(Br)nc1)=O c1(C(=O)NC(C)(C)CCNC(C2CCOC(=O)CC2)=O)ccn2cncc2c1 c1(C(=O)NC(C2CCCN2C(=O)CC2COC(C)(C)CO2)C)ccnc2c1CCO2 C(C1OCCc2sc(I)cc21)NC(=O)C#CC1CC1 c1(N(C)C)ccc2c(c1)CN(C(c1ccc(Br)nc1Cl)=O)C2 CC(F)(F)CCC(=O)NC1CN(C(C2CCCCCC2)=O)CC1CO O(NC(=O)C(CCC1CC1)NC(=O)CCCC1CCC1)CCCC C(=O)(CC(C)N(C(=O)CSCC(C)C)CCC)N(CCC)CCC CCCC(CC(=O)N(C)Cc1nnnn1C)NC(=O)C(C)SC(C)C C1(N(C(COCCC(C)C)=O)C)CCN(C(c2cn3ccnc3s2)=O)CC1C Cc1c(F)cccc1S(=O)(=O)N1CCC(NC(c2ccc(F)cc2O)=O)C(F)C1 N1(c2n(CCCOC)c(Cc3ncc(Cl)n3C)nn2)CCC2(CCCOC2)CC1 N1(C(C2CCCC(C)C2)=O)CCC2(CCN(C(C34CCC(C3)OC4)=O)C2)C1 C1(CC(=O)NC(C2CN(C(C(CC)N(C)C)=O)C2)C)CCN(C)C1=O C(CS(=O)CC(F)(F)F)COC(N1CC(n2c(C(=O)OCC)ccn2)C1)=O C(=O)(N=c1ccn(CCCOc2c(OCC(F)(F)F)cccc2)[nH]1)CCN(C)C C1(C)(NC(C=C(CC)CC)=O)CCCCC1C(=O)NCCC1CC1C c1(C(=O)OC)ccc(CNCC(n2cc(CC(C)C)nn2)C)s1 c1(C(N(CCNC(C(CC)=CC)=O)CC2CC2)=O)ccc2cc[nH]c2n1 N1(C(C2CC(C)(C)OC2)=O)CC2(C1)CN(C(=O)CCc1ccccc1F)C2 c1(C(=O)NC2CCCC(NC(CC(C=C)C)=O)C2)cc2c(s1)COCC2 C#Cc1cncc(C(N2CCN(C(C3SCC=C3C)=O)CC2CCO)=O)c1 N1(C(CC(=C=C)C)=O)CC2(CCCC2NC(C2CCCN2Cc2ccsc2)=O)C1 C(=O)(C(C)(C)CS(C)(=O)=O)N(CC(C)NC(c1c(C)nn[nH]1)=O)C c1(CC)nnc(C)cc1C(=O)NC1CCN(C(=O)CN2CC=CC2)CC1C(C)C c1(OC)c(C)cc(C(=O)NCC2CCCC(CN(C(=O)C=CCO)CC)C2)cc1C C1(NC(COCCOC)=O)CCC2(CC1)CN(C(C1CCCCCC1(F)F)=O)C2 C(=O)(C(CO)NC(C1CCCC1)=O)NCCN(C(=O)CC(C1CC1)C1CC1)C Cc1cc(=NCC2CCC3(CCCC3)O2)[nH]cc1S(=O)(=O)N1CCCC(C)CC1 N1(C(COCCSC)=O)CC(NC(=O)COCC(F)(F)C(F)F)C2CC12 N1(C(C(C(C)C)(C)O)=O)CCC(NC(C2CC3(CCCC3)CO2)=O)C(C)(C)C1 N1(C(CCCNC)=O)CCOC2CCN(C(C3(C)CCN(CC(=O)O)C3)=O)CC12 Cc1cc(C(=O)NCc2ncoc2C2CN(C(c3cnncc3C)=O)C2)sc1C N1(C(CNS(C)(=O)=O)=O)C(CNC(=O)CC23CCC(CC2)C3)CC2COCC12 CC1CCC(CNC(=O)Cc2cnnn2C)N(C(c2ccc(F)cc2F)=O)C1 C1(C(=O)NCCCCOC)(CF)CCN(C(=O)C(C)COC(C)=O)C1 C=CCC(C(=O)NC1CCC(N(C)C(C2COCCO2)=O)CC1)C(C)(C)C C1(C(=O)NC2CC(CCNC(c3c(C)noc3)=O)C2)CCOCC1(C)C C1(C(=O)NC(C2(O)CN(C(C3=C(C)CCC3)=O)C2)C)CCc2cn(C)nc2C1 C(=O)(C(F)(F)C1CC1)NC(C1CCOC1)CNC(CCNC(C1CCC1)=O)=O CC1(O)CCCN(C(=O)CC2C(NC(c3cnsc3)=O)CC2O)C1 C(=O)(C1Cc2ccccc21)N1CCCC(NC(CCC2C(C)C2)=O)(CO)C1 c1(OC)nc(C)ccc1C(c1nnnn1C1COC1)Nc1cc(C)sc1C C1(NC(c2c(O)ccc(OC)c2)=O)COC2(C1)CN(C(C1CC1(C)C(F)F)=O)C2 N1(C(CC=CC(C)(C)C)=O)CC(C(=O)NCC(c2nccs2)C)C2(CC2)C1 c1(C(=O)NCC(=O)NCC(C2CC2)NC(=O)Cc2cnccn2)cccc(O)c1 C1(NC(c2c(COC)noc2)=O)CC1C1CCCN(C(C2(C)CCCO2)=O)C1 c1(NCc2cncc(N=[N+]=[N-])c2)ccc(NC2CCc3ccccc32)c([N+](=O)[O-])c1 Cc1ncc(CCC(=O)NCC(C)(CO)NC(=O)C(F)=CC2CC2)s1 N1(CCC(N2CCOC(CCNC(C3CC(F)C3)=O)C2)=O)Cc2ccccc2C1 Cc1cn2cc(NC(C3CC3NC(c3nc4ncccn4n3)=O)=O)ccc2n1 c1(C(=O)Nc2ccn3ncnc3c2)[nH]nc2ncc(-c3cccnc3CO)cc12 c1(NCC=C)nccc(C(=O)OC)c1[N+](=O)[O-].C12CC1CN(C)C2=O N1(C(CCN(C(=O)CCOC2CC2)CCC)=O)CCC(n2cncn2)C1 CCCCC(C)CCC(=O)N1CCC(N(C)C(c2ccc(Cl)cc2Cl)=O)C1 CC1CCOC(C(N2CCC(C(C)(C)C)(CNC(=O)C(C)(F)F)C2)=O)C1 c1(C(=O)NC2C3CN(C(CN(C4CCCC4)C)=O)C2C3)cnc2ccc(Cl)cn12 c1(OC)ccc(C(C)C(=O)N2CC(C(C)NC(c3cc(F)c[nH]3)=O)C2)cc1 C1(NC(C2CC3CC(O)C(C2)C3)=O)CCS(=O)(=O)C12CN(C(=O)CCCF)C2 c1(CC(=O)NCC(CC=C)NC(=O)C(C)CCC)ccc(C)c(Br)c1 C12(CNC(c3c(C)nc(N(C)C)s3)=O)CCC(CC1)N2C(=O)C(C)(C)NS(N)(=O)=O C1(SCC(=O)N(C(C)C)CCN(C(=O)C(C2CCOCC2)O)C)CCS(=O)(=O)C1 c1(C(N2CCC(OCCCNC(=O)C3=CSCS3)CC2)=O)ccn2cccc2c1 c1(C(N(C)C)=O)cccc(C(=O)NC2CN(C(c3cnc(N)cn3)=O)C3CC23)c1 N1(C(c2c(CSC)cccn2)=O)CCC(NC(=O)C=Cc2nc(C)cs2)C(C)C1 C1(NC(c2cncc(C(C)C)c2)=O)CSC12CN(C(=O)C(C1CCCCC1)F)C2 O=C1CC(C(N2CC(CO)(NC(=O)C(C3CC3)C3CC3)C2)=O)Oc2ccccc21 c1(OC)cccc(C(=O)NCC2CCCN(C(=O)C3=C(C)CCC3)CC2)c1F C1(n2cc(CC=C)nn2)CC2CCC1(NC(c1ccc(F)cc1)=O)C2 N1(C(C2(CC)CCCO2)=O)CCC(C(=O)NCC(c2cccnc2)O)C(C)C1 c1(CN(C(C(C)(C)NCC=C)=O)C)cccc(Br)n1 N1(C(CCC=C(C)C)=O)CCC(C)(C)C(C(=O)NCCN(C)C2CC2)C1 N1(C(C(C)OCCC(C)C)=O)CC2CC1C2NC(c1nccn1C)=O c1(CC(=O)NCCC(CNC(CCC)=O)O)c(C)cc(N(C)C)cc1C C1(NC(C(CCOC)C)=O)CC(C)CN(C(=O)Cc2ccsc2Cl)C1 N1(CC(C2CC2)OCC)CCC(CC(N2CCSCC2)=O)C1 c1(C(C)(C)C)ncnc(C(F)(F)F)c1Br.c1(C(C2CCCNC2)N)ncc(Br)cc1F c1(COC2CC(C(=O)OC)C2(C)C)cc(C(F)(F)F)ccc1Cl C1(OC)CC2CC(COc3cc(OC(C)=O)ccc3OC(C)C)CC12 N1(C(c2c(C)nn(CCO)c2)=O)CCC(C2CC2NC(c2nnsc2C)=O)CC1 C1(C(=O)NCCCC(C)NC(c2ccn(C(C)(C)C)c2)=O)CC2CCC2C1 c1(NC(C23C(CN(C(CCOC)=O)C2)C3)=O)ccc(Br)c(Cl)c1 C12(C(=O)OC)COCC1CN(C(N1CCC(Oc3ccc(C#N)cc3)CC1)=O)C2 c1(C(=O)NCCCCN(C(=O)CCSCC(N)=O)C)ccc(C(F)F)cn1 c1(C(N2CC(C(C(=O)N(CC(C)O)CCF)O)C2)=O)sccc1F N1(C(C(C)(C)OC)=O)CCCC(F)(CNC(c2cn(C(C)C)cc2C)=O)C1 CC1CCC(C(=O)NC2(C3CC3)CC2)N(C(C2CC=CCC2)=O)C1 c1(C(N(CCN(C(Cn2c(C)cnc2)=O)C(C)C)C)=O)ccc2c(c1)CCCS2 C1(OC)CN(C(C2CCCC2CF)=O)CCC1NC(=O)CCNC(=O)C(C)(C)C C(=O)(CCCCCCN=[N+]=[N-])NCC1CCN(C(C2CC3(ON=C(C)C3)C2)=O)C1 Cc1cc(C(F)(F)F)sc1C(=O)N(CCNC(=O)C(C1CCCCC1)O)C(C)C c1(N2CCC(C)C2CNC(c2cc3n(n2)CCCO3)=O)cnc(C#N)c(C#N)n1 N1(C(Cc2cccc(OCC)n2)=O)CCC(NC(c2csc(C)n2)=O)CC1C c1(C(=O)NC(C2(O)CN(C(=O)CC3CCNC(=O)C3)C2)C)cc2c(s1)CCOC2 c1(C(N2C(C(=O)NCC3CCOC3)COCC2)=O)cccc(F)c1F c1(COC)ccc(F)c(C(N2CC(C)C(C)(C(=O)OC)C2)C(=O)NCCSC)c1 Cc1cc(C(=O)NC(CO)C(C)NC(C2CCn3nnnc3C2)=O)c(C)cc1Cl C1(NC(c2c(OC)cc(C)s2)=O)CCCCN(C(=O)C(C)(O)c2ccccn2)C1 C1(C(=O)NCc2c(C)cncc2)CC2C=CC1N(C(=O)C=Cc1cncn1C)C2 C(=O)(C(C#N)C(C)(C)C)N1CC(C(=O)NC2CC(OCC)C2)C(C)C1 c1(C(N2CC3C(C(=O)NCCN4CCOCC4)C3C2)C)n[nH]c2ccccc12 C(=O)(CCC(=O)NCCNC(C)=O)N(CC(=O)OC)CC#C CCCCCCC(=O)N1CCC(NC(=O)C(CC)NC(N)=O)C1 C1(CC(=O)NCC2N(C(c3c(C)cno3)=O)CCN(C)C2)Cc2ccccc2N1 c1(N2C(C(C)(C)NC(C3(c4cccnc4)CCC3)=O)CCC2)ccc(C#N)nc1 Cc1ccc(NC(=O)CC2CCCC(C#N)C2)cc1O c1(CC(N2C(C(=O)NCC(CC)N(C)C)CC2)=O)cc(C)on1 c1(C(CN2CCN(C(C(CC(=O)O)C(F)F)=O)CC2)=O)ccc2c(c1)OCCO2 C1(CNC(C(C(C)O)NC(c2cc(Cl)ns2)=O)=O)COCC(=O)N1C N1(C(c2c(CCC)[nH]cc2)=O)CCC(O)(CNC(c2cccc(C3CC3)c2)=O)C1 c1(C(=O)NCC2C(NC(=O)CCSc3ccccc3Cl)C2)ncc2ccccn12 CCC(O)C(C)(C)C(=O)NCCc1cc(C(=O)NCCc2ccc(C)s2)no1 c1(OCCN2c3ccc(cc3)C2C(=O)NC)cc(C)ccc1Cl.C(C)(C)(C)SC c1(NC(C2CC(=C)CN2C(c2ccc(OC(F)(F)F)s2)=O)=O)c(C)cccc1Br c1(C(=O)NC23CCN(C(c4ccc(Cl)cn4)=O)CC2C3)ccnc2ccccc12 C1(C)(C(=O)NC(C)C)CCCN1C(=O)CCNC(N)=O N1(C(CC2(C)N(C(C3CC(O)C(F)C3)=O)CC2)=O)C(CO)CCC12CCC2 C1(C(N2C(CNC(c3cc(O)ccc3F)=O)CCC2)=O)CCC12CCOCC2 Cc1noc(C)c1C=CC(=O)NC1CC(C)CN(C(c2c[nH]cc(F)c2=O)=O)C1 c1(CNC(C(c2n(C)ccn2)(F)F)=O)ccc(CCNC(c2ccon2)=O)cc1 C1(NC(CSc2cc(C)on2)=O)CN(C(=O)C(C)SCC2CCCO2)CC1C N1(C(C2CC(C)N2C(c2ccc(=O)n(C)c2)=O)=O)CC(CO)CC1(C)C N1(C(C(CC)c2cccnc2)=O)CCCC(N(C)C(c2ccc(N)cn2)=O)C1 c1(C(N2CCN(C(c3occ(C)c3)=O)C(CO)C2)=O)cc2c(Cl)cccc2[nH]1 CC1(C)COCCN(C(=O)C(c2cccnc2)NC(=O)C(C2CCCCC2)F)C1 CC1CC(NC(C2CC3CCC3C2)=O)CN1C(=O)CCCOC(C)(C)C CCC(CC(F)F)C(=O)N(C(CNC(c1cnc2c[nH]nc2c1)=O)C1CC1)C C1(O)(CCNC(C(C)N(C(C)=O)C)=O)CCN(C(=O)CCC2OCCO2)CC1 Cc1nccc(Cl)c1C(=O)NC1CCN(C(=O)C(=O)NC2CC2)CC1CO N#Cc1cc(C(=O)NCC23CC2CN(C(=O)C2=C(Cl)CC2)C3)co1 CC1=C(C(=O)NCC2(F)CN(C(=O)Cc3scnc3C)C2)C(C)(C)CCC1 Cc1cc(C)c(C(=O)NCCCCNC(=O)CCc2ccccc2)cc1N Cc1cc(NC(=O)NC(CC2CCCCC2)CO)ccc1N(C)C Cc1c(C(N2CCC(N(C(=O)CCC(C)N(C)C)C)CC2)=O)ccc2n[nH]cc12 N1(C(C(C)NC(c2ccc(C)cc2)=O)=O)CC2CC(C1)C2NC(=O)C#CC(C)C c1(C(=O)NC2CC(C)CN(C(=O)C=CC3CCC3)C2)n[nH]c2ccc(F)cc12 N1(C(CCC2(C)CC2)=O)CCCCCC1CNC(c1ccc(F)cc1C(F)F)=O c1(C(=O)OC)ccc(N2CCC(O)C(C)C2)c([N+](=O)[O-])c1 C1(CNC(C2CC(OC)C2)=O)(NC(C2(C)CC2(F)Cl)=O)CCCCC1C CC(C(=O)NC(C1(O)CCN(C(=O)Cn2nnc(C3CC3)n2)CC1)C)C(C)(C)C c1(C(N2CC(C(=O)NCCOC(F)(F)F)NCC2)=O)cc(I)ccc1Br c1(NC(N(CC(C)(C)CCO)C)=O)cccc2c1CCCC2=O CC(C(=O)N1CC(NCC2CCCC2)C1)NC(C1CCCC1)=O c1(C(=O)NC(CC)CN(C(=O)CCC2CCCCO2)CC)noc2c1COCC2 C12(C(=O)NCC#CC(=O)NCC(F)(F)F)CC1CNC2=O N1(C(c2nc(CNC(c3cc(C#N)[nH]c3)=O)oc2)=O)CC2(CCCC2)C1 C1(C(=O)NC2CN(C(c3c(C)ncc(C)c3)=O)CC(C)C2)CCn2nnnc2C1 c1(C(=O)NCC2CCC(NC(C(C)S(C)(=O)=O)=O)CC2)cc(F)c(F)c(F)c1F C1(C(=O)NC(C(=O)NCC)CC)CCCN(C(c2ccn(C)c2C)=O)C1C N1(C(C(CCC)=CCC)=O)CC2CCN(C(=O)C(C)CCCC)C2C1 N1(C(CCSCC)=O)CC=CC(NC(C2CCCCN2C)=O)C1 C=CCCCC(=O)NC(c1ccc(F)cc1)CNC(=O)CN(CC)CC C1(CNC(C2C(COC)C2)=O)CN(C(c2c(F)cncc2Cl)=O)CC2(CCC2)O1 N1(C(C(C(C)(C)C)C#N)=O)CC(C2CCCN(C(c3cnc4n3CCS4)=O)C2)C1 c1(OC)ccc(C#N)cc1CNC1(c2ccccc2C#N)CC1 c1(CCC(=O)NC2CN(C(C(=O)NCCNC(N)=O)=O)C2)ccccc1[N+](=O)[O-] C(=O)(CCC(C)(C)C#N)N1C(C(N(CC(=C)C)C)=O)CCCC1 c1(NC(C(N2C3CN(C(C4CC(OC)C4)=O)C(C3)C2)=O)=O)ccc(C#N)c(Cl)c1 c1(C(C(F)(F)F)NC(Cn2c(C)cc(CO)n2)=O)ccnc2ccccc12 C1(NC(c2cc3scnc3[nH]2)=O)CC2CCC1CN2C(=O)Cc1ccc(F)nc1 C(C(C)(C)CC(=O)NC1CCC(NC(C2CCCCC2C(=O)NC)=O)C1)OC C1(S(C)(=O)=O)(C(=O)OC)CC(C(=O)Nc2ccc(Br)cc2Br)CC1 N1(C(CC(CCC)CCC)=O)CCC2CN(C(=O)C=Cc3cncs3)CCC2C1 C1(CNC(C(c2cccc(Cl)c2)C)=O)CN(C(c2cc[nH]c(=N)c2)=O)CCO1 CC1(C(N2CC(O)(CNC(=O)CC3(c4ccon4)CC3)C2)=O)CC(F)(F)C1 c1(C(=O)NCC2CN(C(c3c(C)onc3)=O)C(C)C2)ccc(=O)n(C(C)C)c1 C1(C)(CNC(COC2CN(C(C)=O)C2)=O)CN(C(c2ccon2)=O)CC1C c1(CN(C(c2ccccc2)C(C)=O)C(N)=O)cn(C(C)C)nn1 Cc1cc(Br)cc(Cl)c1CN1CCCC1C(=O)NCC(C)C c1(C(N2CC(C)C(CNC(=O)CCc3ccoc3)C2)=O)cccc2nccnc12 N1(C(c2nccc(C)c2)=O)CCCC2C1CCN2C(c1cc[nH]c1C1CC1)=O N1(C(CC(CC)CN(C)C)=O)CCCc2c(CC)ccc(C)c21 c1(CC(=O)NCC2CCN(C(=O)Cn3cnnn3)C2)cc2ccccc2c(=O)o1 C(=O)(C1=CC2CCCCC12)N(CC(CC)NC(c1nnsc1N)=O)CC N1(C(CN(CCCCCC)C)=O)CCC(C2CCN(C(=O)CCOC3CC3)C2)C1 C1(NC(=O)CCCC2CCC2)COC2(CCN(C(=O)CCCCC(F)(F)F)C2)C1 C=CC1CCN(C(C2CCCN(C(C3CCC3C#N)=O)C2)=O)C1 C(C(COC)C(=O)NCCCCCCNC(C1CCOC(C(C)C)C1)=O)OC c1(CN2CC3CCN(S(=O)(=O)CCCCl)C3C2)cccc2nscc12 C1(C(N2CC(C(N)=O)(CNC(C(n3ccc(C)n3)(C)C)=O)C2)=O)CC2(CC(=O)C2)C1 C1(C)(CC)CC(C(N2CCN(c3cc(N)nc(SC)n3)CC2)=O)CCO1 Fc1cccc(Cc2noc(CNCC(F)=CC=Cc3ccccc3)n2)c1 c1(CNC(c2cc3ncn(C)c3s2)=O)nc2c(s1)CC(c1ccccc1)CC2 c1(C(=O)NC23CC(CC)(C2)C3)ccc(CNC(=O)CCN2CCC(C)CC2)nc1 Nc1nc2c(cc1C(=O)N(CCNC(C1CCSCC1)=O)C1CC1)CCCC2 C1(C(C)C)CN(C(C2CC23CC(C)(C)C3)=O)CCN1C(c1ncc(F)cn1)=O CC(CC(=O)NCCCCC1CN(C(C2CC3(CCCO3)C2)=O)C1)CC(C)(C)C C(CC(C)(C)C)(C(F)(F)F)NC(c1cccc(C(C)O)n1)=O c1(C(N2CCC2CO)=O)cnc2c(-c3ccc(F)cc3F)cnn2c1 C(=O)(CS(=O)(=O)C1CCCC1)NC1CCN(C(c2c(C)n(C)cc2)=O)CC1 C1(NC(C(C)n2ccnn2)=O)CCCC1CN(C)C(c1csc(O)n1)=O c1(CN2CC3N(C(C4(OC)CCC4)=O)C3C2)nccc2ccccc12 S(=O)(=O)(c1c[nH]c2cccc(F)c12)NC(C)(C(=O)O)C1CCOC1 c1(C(=O)NCC(C)N(C(=O)C(C)NC(N)=O)CC)nn(C)cc1C C(C(CNC(C12CC(F)(C1)C2)=O)CO)NC(C1(COCC)CC1)=O c1(C(N2CCC(N(C(=O)Cc3sc(O)nc3O)CC)C2)=O)cc(Cl)c(Cl)cc1Cl c1(-n2c(-c3ccc(C(F)F)nc3)nc(C(C)OC)n2)cc(F)c(F)c(F)c1 C1(C2(NC(c3cc(C)no3)=O)CC2)CCCCN1C(c1ccc(CO)o1)=O N1(C(c2n(C)ncc2Cl)=O)Cc2ccccc2C(NC(=O)CC(C)(C)C#N)C1 c1(OCC)ccc(F)c(C(=O)NCC(C2CC2)NC(C2(CC3CC3)CC2)=O)c1N C1(NC(CC(=O)NC)=O)CN(Cc2cc(OC)nc(C(F)(F)F)n2)CCC1C C1(C(N(CCC(=O)NC(C)CN(C)C(C)C)CC=C)=O)CCC2(CCC2)O1 c1(OC)cc(Br)cc(S(=O)(=O)CC(=O)N2CC(C)OC(C)C2)c1 CCC(CNC(C1CC(NC(C2CCCC2)=O)C1)=O)CC(C)C c1(C(C)C)ncc(C(=O)NCC(C)NC(C2(CS(C)(=O)=O)COC2)=O)n1C C(=O)(NN1CCCC1C(=O)NCCCC1CC1C)c1n[nH]c(C)c1O c1(OC)cccc(NC(=O)C(c2cccc(F)c2)N2CCC(F)(CF)C2)c1 c1(C(N2CC(CC)C(NC(=O)Cc3cccnc3)C2)=O)n[nH]cc1[N+](=O)[O-] C(C(C)CC(C)C)(c1nnnn1Cc1nnn(C)n1)NCC(=O)OCC=C c1(C(C(=O)NC(CC)C)N(C2CCOCC2C)C)nc(C2CC2)n(C)n1 N1(C(COCCCCC)=O)CCC(C(C)(C)NC(=O)COCC)CC1 N1(C(COCC)=O)CC2OCCN(C(c3cncc(COC)c3)=O)C2C1 c1(CC(=O)NCCN(C(=O)CCc2cn[nH]c2)CCC)ccc(OCC#N)cc1 c1(CC)nnsc1CNC(C1CC2CC2C1)c1nnnn1C(C)(C)C N1(C(C(CC)=CC)=O)CC2CC(C1)CN(C(=O)CC(O)C1CCCC1)C2 C1(CC#N)CCC(C(=O)NC2CCCC(C(=O)NC3CCCCC3CO)C2)CC1 c1(C(C)C)ncsc1C(=O)NCC1CC1CNC(=O)COC1CC(F)(F)C1 N1(C(CCOC(C)=O)=O)CCOC2(CCC(NC(C3(C(C)(F)F)CC3)=O)CC2)C1 C1(CC(=O)NCC(O)CF)C2CCCC2N1C(=O)C=Cc1ccco1 n1(CC(=O)NCCN(C(c2ccnc3[nH]ncc23)=O)CC)ncc2cccnc12 c1(C(C(=O)NC)N(C)Cc2snnc2C)cc(C(=O)OC)c(C)o1 CC1(C)C2CCC(CC(=O)NCC(C)(O)CNC(=O)C=C3CCC3)C1C2 Cc1nc2ccc(C(=O)NC3CC(O)CN(C(=O)Cc4cnnn4C)C3)cn2n1 c1(CC(=O)N(C2CCN(C(=O)C3=COCC3)CC2)CC)cc(C)cc(F)c1 c1(CN2CCC(NC(c3ncc(Cl)cc3Br)=O)C2)cc2cc[nH]c2cn1 C1(NC(C(C)OC2CCCC2)=O)CCCCCC1NC(C1COCCN1C)=O Cc1c(C(=O)NCC2(NC(=O)Cc3cnns3)CCC2)cncc1Br C1(NC(C2(C#C)CN(C(c3cc(C)oc3CC)=O)C2)=O)CCCCNC1=O C(=O)(CCCCC1CC1)NC(C(N1C(CCC)CCC1)=O)Cc1ccco1 NS(=O)(=O)c1ccc(C(N2CCCC23CCCN(C(=O)C2CC2)C3)=O)cc1[N+](=O)[O-] C1(C2CCN(C(=O)C(c3ccnn3C)O)C2)(NC(C2CC(SC)C2)=O)CC1 N1(C(c2ncn(C(C)(C)C)c2)=O)CCN(C(C2CCCC2)=O)CC(CO)C1 c1(OC)c(C(=O)NCC(C(C)(C)C)NC(C2C(Cl)(Cl)C23CC3)=O)csc1Cl C(CN=C(NCC1(c2cccc(Cl)c2)CCCC1)N1CC(F)(F)C(F)(F)C1)OC C(C(CO)(CO)NC(=O)CC1CCCCN1C)N(C(C1(CC#C)CC1)=O)C C1(=CC(=O)NC2CCN(C(CC(=C=C)C)=O)C(C)C2)CCOc2ccccc21 N1(C(C(C)(CSC)NC(C=CC(CC)C)=O)=O)CCC(CO)C(O)C1 C=C(C)C(C)(C)C(=O)NC1C=CC(CC(N2CCC(Cc3ccccc3)C2)=O)C1 C1(NC(C(CO)N(C)C)=O)CCN(C(c2cccn3cnnc23)=O)CCC1(F)F C1(CNS(CC2(SC)CCC2)(=O)=O)(COC(C)(C)C)CC(C(=O)O)C1 C(C(C)CC(=O)NC1CC(NC(=O)CCCc2nc(C(C)C)no2)C1)OC C(=O)(C(CC1CCCC1)OC)N(CCOCCN(C(COC)C)C)C Cc1cc(C(N2CCCCC2C2CCCN(S(C)(=O)=O)C2)=O)oc1C CC1=NC(C)(CNC(c2oc(CNC(=O)C(C)c3cccs3)cc2C)=O)CS1 C(C(C)C(C)C(=O)N1CCCC1CN(C(=O)C(C1CCCO1)C1CC1)C)OC CC(C)CC(O)CC(=O)N(CCCCC(=O)NC1C(C)CCC1C)C c1(C(=O)NCCC(C)NC(CCOC(CC(C)C)C)=O)cc(Cl)c([N+](=O)[O-])[nH]1 N1(C(c2cc(CC(C)C)on2)=O)CCCN(C(=O)CCC2CCCC(O)C2)CC1 C12(C(=O)NC3C(CNC(=O)CCc4cc[nH]n4)CCC3)CCCC(=O)N1CCC2 c1(OC)csc(C(=O)NCCn2cc(CO)nn2)c1NC(=O)CN1CCC1C c1(C(N2CC(N(C(C(n3cc(Cl)cn3)C)=O)C)C2)=O)ccc2sccc2c1 N1(C(c2n(CC(C)C)ncc2)=O)CCC(N(C(=O)C(C)OCC2CC2)C)CC1 N1(C(Cc2ccc(C)cc2F)=O)CCC(NC(=O)C(C)CO)CC(C)(C)C1 C1(CC(=O)NCC)CCCN(C(=O)CNc2ncccc2C(=O)OC)C1 C1(C(=O)NCC=C=C)CCCCN1C(=O)Cc1cnns1 N1(C(C(F)OC)=O)CCN(C(C2C3CCC2(c2ccn(C)n2)C3)=O)CC1C Cc1ncccc1C(=O)NCCCCN(C(=O)C(F)CC1CCCC1)C CC(CC(=O)NCCNC(C12CC(F)(C1)C2)=O)N(C)C(=O)OC(C)(C)C N1(C(c2c(C)cn(C)c2)=O)CCN(C)CC1C(=O)NCCc1ncoc1C N1(C(c2cc(C)c(F)cn2)=O)CC2CCCC2(NC(C2CCCO2)=O)C1 C(=O)(C1CCCc2ccnn21)NC(CC)CNC(c1cc(F)c(C#N)c(F)c1)=O c1(C(N(C2CCCN(C(=O)CC3C=CCCC3)C2)C)=O)cc(O)c2ccoc2c1 N1(C(=O)OC(C)(C)C)CCCCC(NCC(c2ccc(Cl)cc2)(C)C)C1 O=S(=O)(CC1CCOCc2ccccc21)N1CC2(CC2)c2ccccc21 CC1(C)CSCCN1C(c1occc1Br)C(=O)NCCOCC1CC1 C1(CC)CCCN(CC(=O)NC2(C)CN(C(C3CC3CC(C)C)=O)C2)C1 c1(C(=O)NCCN(CCN2CC3CC3C2)C2CC2)cc(=O)c2ccccc2o1 C(=O)(C1=C(C#N)CCC1)N1C(CNC(c2c(C)onc2)=O)C(C)CC1 C(C(=O)Nc1cnn(CCF)c1)(C(C)OC)NC(C1N(CCC)CCC1)=O N(S(=O)(=O)N1CCC(C#N)C1)Cc1c(C)nc(-c2ccccc2)s1 CC1CN(C(=O)CC(=O)NC2CC2)CCN1CC(F)(F)F c1(N2CC=CC(OC)C2)nc(N2CC3CN(C(C)C)CC3C2)nc2ccsc12 CCCCCCn1nnnc1C(CCOCC1CC1)NCC(C)(C)N1CCCC1 N1(C(C2C(OC)(OC)CC2)=O)CCCCC1CN(C)C(c1sc(F)cc1Cl)=O Cc1cncc(C)c1C(=O)N(CCCCNC(C1CN(C)CC1C)=O)C CCCCC(C)(F)C(=O)NC1CN(C(c2ccc(C#N)cn2)=O)CC1SC c1(C(=O)NC23CN(C(C4(Cl)C(C)(C)C4)=O)C(C2)C3)cc2n(n1)CCNC2=O Cc1ccc(C(N2CC(OCC(=O)NCCCC3C=NNC3=O)C2)=O)nn1 C1(C(=O)NCCCC(C)NC(c2cc(C3(C)CC3)on2)=O)CCCC2CC12 Cc1cc(C(=O)NCc2ccoc2C(=O)NC(C)CC2CCCCC2)cc(C)c1 CC1CN(C(c2ccn(C3CCCCC3)n2)=O)CCC1NC(c1coc(Cl)c1)=O N1(C(CC(=O)N(C)C)=O)CCN(C(=O)C=C2CCC2)CC1c1nccn1C C#Cc1ccc(C(=O)NC23CC(CNC(C4CCC(F)(F)C4)=O)(C2)C3)o1 CC(C)CC(C)(CNC(=O)C(C)CF)NC(c1ccc(Cl)cc1C(F)F)=O CC(CC1CCC1)C(=O)NCCCOCCNC(c1sccc1SC(F)F)=O C1(C(C)NC(=O)OC2CN(C(=O)CSCC(N)=O)C2)CCN(C=O)C1.C(C)(C)(C)O N1(CC(=O)N(C2CCC(NC(=O)COc3ccsn3)C2)C)C(=O)NC(C)(C)C1=O c1(C(N2C(C(C)NC(C(C)(C)OC)=O)CCC2)=O)cc(F)cc(F)c1F c1(CN2C(CNC(=O)CNCc3cccs3)CC(F)C2)ccc(Br)cc1I N1(C(CCCCC=CC)=O)CC(C)(C)OCC1CNC(=O)C(C)CSC C12(CNC(C3CC(CCC)OCC3)=O)CN(C(C3CC=CCC3)=O)CC(F)(C1)C2 c1(C(N2CCC(C(=O)OC)(OC)C2)C(=O)NC)ccc(-n2ccnc2)cc1 C1(C(=O)NCC2(CN(C)C(C3CCS(=O)(=O)CC3)=O)CC2)(OC)CCC12CCC2 C(=O)(C(C)(C)C(C)C)NC1CCC(N(C(c2cn(CC(C)C)nc2)=O)C)C1 c1(CC)ncc(C(=O)NC2COCC2CNC(=O)C(C)(C)n2ccnn2)c(O)n1 c1(CN(C(=O)C(C2CC2)N(C)C(=O)OC(C)(C)C)CC)ccccc1O c1(C(N(C2CN(C(C3CCS(=O)(=O)N3C)=O)CC23CC3)C)=O)c[nH]cc(Cl)c1=O CC1CCCn2cc(C(=O)NC34CC(CNC(c5coc(CO)c5)=O)(C3)C4)nc21 c1(OC)ccc(F)c(C(=O)NC(C)(CNC(C2(O)CCOCC2)=O)CC(C)C)n1 N1(C(CCC)C)CC(C(=O)NCC2CC(NC(=O)CCOC3CC3)C2)CC1=O Nc1cc(Cl)nc(Cl)c1C(=O)NCCN1CCN(C(C2CC(F)(F)C2)=O)CC1 C1(C(=O)NCCN(C(=O)CN2CC=CC2)Cc2ccccc2)COCCO1 CCCCCCCC(=O)N1CC2CC(C(=O)Nc3cnc4c(c3)CCC4)C(C2)C1 c1(CC)nc(C(=O)NCC2CC2CNC(=O)CC2CCC2)c(N)s1 N1(C(c2c(CC)nns2)=O)CC2C(CNC(=O)C(CC)c3cccnc3)C2C1 C1(CNC(CS(=O)(=O)NC)=O)C(C)CCCN1C(=O)Cn1ccnn1 N1(C(C(c2cccc(C)c2)C)=O)CCCCC(NC(c2ccc(F)c(N)c2)=O)C1 c1(C(N2CC(C)CC2C)C(=O)NCCC)cncc(C)c1 CS(=O)C1(CNC(c2nnnn2CC2CCOCC2)c2ccsc2)CC1 n1(CC=C)cc(C(=O)N(CC(C)N(C(=O)C(C)NC(C)=O)C)C)nn1 c1(C(N2CCC(NC(c3cc(O)cs3)=O)C2)=O)cccc(N2CCCNC2=O)c1 N1(C(c2cnc(C)s2)=O)CCC2CCN(C(=O)CS(N)(=O)=O)CC12 c1(CC(=O)NC23CC(NC(C=COCC)=O)(C2)C3)cnccc1C Cc1ccc(=O)n(CC(=O)NCCN(C(C2SCCC2C)=O)CC2CC2)n1 C12(CNC(C(CC)OC)=O)CCCC(CN1C(=O)Cc1nnsc1Cl)C2 C1(C(=O)NC2CC3CC(C2)N(C(=O)C2=CCOCC2)C3)CCC2(CC1)OCCO2 Cc1cccc(C(C)C)c1C(N1CCCC1CNC(C1COC(=O)N1C)=O)=O C1(C(N2C(C(N3C(C)(C(=O)NC)CC3)=O)CC2)=O)COCC1(C)C N1(C(C=Cc2occ(C)n2)=O)CC2(CC(NC(c3cn(C)cc3C)=O)CO2)C1 C1(C(=O)NCCN(C(c2cccc(OC)c2C)=O)C(C)C)CCN2CCOCC12 CC1(C)CCN(C(=O)Cn2cnnn2)CC1C(=O)NCCCCC1CCCC1 c1(OC)ccc(C(=O)NC(C(=O)N(C)C2CC2)C2CCOC2)s1 C1(CNC(CN2CCC(OC)C2)=O)CN(C(C2(CO)CCCO2)=O)CCCO1 C(C(O)(CNC(=O)CC1C2CN(C(=O)Cc3cncnc3O)CC12)CO)OC N1(C(c2c(C)scn2)=O)CCCC(F)(C(N2CCC(O)CC2C2CC2)=O)C1 N1(C(COCC=C)=O)CCC2OCCN(C(=O)CCn3cccc3)C2C1 c1(SC)nc(C)cc(=NC(C(C)NC(c2ccncc2)=O)C(C)C)[nH]1 CC1CC2CN(C(C3(C)CC(O)CN3C(c3cc(O)ncc3F)=O)=O)CCN2C1 CCCC(C)CC(=O)NC1CC2CC1N(C(c1cc(C(F)F)n(C)n1)=O)C2 C12(NC(c3cn(CCC)nc3)=O)CCCN(c3ccc(C#N)nn3)CC1C2 CC1c2cccc(Br)c2CCN1C(=O)N=c1ccn(C(C)(C)C)[nH]1 C(=O)(CCCCCN(C)C)N(CC(CC)NC(c1oc(CC2CC2)nc1C)=O)C C1(C(N(C)CC2COCCN2C(=O)CCCc2cccs2)=O)CCCCS1(=O)=O N1(C(c2cc(OCC)no2)=O)CCN(C(C2(OC)CCSC2)=O)CC1C C1(NC(=O)Cc2c(F)cccc2Cl)CC2CC(C1)N(Cc1noc(C3CC3)n1)C2 N1(C(c2c(CC)ocn2)=O)CC(C(N2CCC2C(C)O)=O)CCC1(C)C Cc1cc(C)c(C(=O)NC2CC2NC(=O)C(c2ccccc2F)N(C)C)c(O)c1 N1(c2nc(CC)nc(Cl)c2C)CC2(C)CN(C(C3(CN(C)C)CC3)=O)CC2(C)C1 N=c1nc2c(c[nH]1)CC(C(N1CC(NC(=O)C(F)=CCCF)C3(CC3)C1)=O)CC2 Cc1cc(CNC(C2NCC3CC23)=O)nc(O)n1 C(=O)(C(C(=O)N(CCCCNC(=O)CC1(OCC)CCC1)C)OC)OCC c1(C(=O)NCC(C(C)C)NC(C=CCCC)=O)ccc(OC)nc1C CCCCCCC(CC)C(=O)N1CCC2(CCN(C(=O)Cc3ccoc3C)C2)C1 c1(C(c2n(CC=C)nnn2)NCCC2CCCO2)c(Cl)nc2sccn12 C1(CN(C)C(C2CCCN2C2CCCC2)=O)CCN(C(C2(C(N)=O)CC2)=O)CC1 C12(C(N3C(C)CN(C(C4CN=C5N=CNN5C4)=O)CC3)=O)CC3CC1C2C3(F)F C1(NC(c2nnn(C)n2)=O)(CNC(=O)Cc2cccc(F)c2)CC2CCC1CC2 N1(C(C2(CC)CCC2)=O)CCN(C(=O)Cc2cc(Cl)cc(Cl)c2)C(C)C1 C(C(CC(=O)N(C(C)CC(C)C)C)NC(=O)C(C)(F)c1ccon1)OC c1(CC(N(C2C(C)CCC2)C(=O)OC)=O)c[nH]c2c(F)cccc12 CC1(C)CCN(C(=O)CCc2cnco2)C(C(=O)NCC2CC2(Cl)Cl)C1 N1(C(C(CSC)(C)NC(=O)CCc2nncs2)=O)CCCNC(=O)C1CC C(=O)(C(F)CC(C)(C)C)N(CC1N(C(CC(C=C)C)=O)CCC1)CC c1(C(N2CCC(C(=O)NC3(C(C)C)CCOCC3)C2)=O)ccc(Cl)cc1Br c1(C(=O)NC2(CNC(C(COC)O)=O)CCOC2)cccc2nc(C)cnc12 c1(OC)cc(OC)cc(C(O)CNC(C2CC3CCC2(N)C3)=O)c1 C12(COC)CCC1CCN2C(=O)CCN(C)C(=O)OC(C)(C)C C1(CC)CN(C(=O)CN(C)C(N)=O)CCC1NC(C1(c2ccsc2)CC1)=O CCCCS(=O)(=O)NC(C)C(=O)NC1CCCCC1NC(C1CC(SC)C1)=O C1(NC(C(=O)NCCOCCCC)=O)CCCN(C(c2cscc2F)=O)CC1 C1(C(=O)NCC2(C(N)=O)CN(C(=O)C3=NOCC3)C2)CN2CCC1CC2 C=Cc1ccc(C(=O)NC2CCN(C(c3[nH]cnc3C)=O)C(C)C2)cc1 CC1CC(C(=O)NC2CC(CNC(=O)C(C)(C)c3ccns3)C2)CCS1 C1(C(N(CCN(C)C(c2c[nH]c(=O)cn2)=O)C)=O)CC(c2ccccc2)=NO1 c1(CC)nc(C(C)C)ccc1C(=O)NC1CC(N(C)C(c2nc(=N)cc[nH]2)=O)C1 Cc1cnc(N)c(C(=O)NCCCN(C(=O)CN2CCC2C)C)c1 C1(NC(c2c(C)snn2)=O)CCCCC1NC(=O)CCOCc1ccccc1 C1(NC(C(c2cncc(F)c2)C)=O)CCN(c2ccnc(CO)n2)C1C c1(C(N(CC(C)NC(=O)CCc2cn(C)nn2)C)=O)cc2cc(F)ccc2o1 c1(OC)cccc(C(N2CCC(C)C2CNC(=O)COc2ccsn2)=O)c1N C(=O)(C(C(CC)CC)OC)NCC1CCN(C(C(CCC)=CCC)=O)CC1O c1(N2CC(CCNC(CCCC3CCCC(=O)N3)=O)C2)ccc(Cl)cc1[N+](=O)[O-] c1(OC)cc(OC)c(S(=O)(=O)NC(C)(CC(=O)O)c2cccnc2)cc1C c1(N2C(c3ccc(C)cc3)COCC2)cc(Br)ccc1S(=O)(=O)NC1CCSC1 NC1CCc2ccc(NC(C3CC(=O)NC(c4ccccc4)C3)=O)cc21 c1(C(=O)NC2CC(=O)N(C3CN(CC(=O)NC4CCC4)C3)C2)cccc(Cl)c1 C(=O)(CCC(C)(C)C#N)N1CC2(C(NC(c3c(C)ncs3)=O)CC2)C1 c1(OC)ncccc1S(=O)(=O)N1CCCC(CCNC(c2cncnc2C)=O)C1 c1(N2C(CCNC(c3cccc(N(C)C)n3)=O)CCCC2)cncc(C#N)n1 C1(N(C(CC)C)C(c2csnc2Oc2ccccc2)=O)CCN(CC)CC1 N1(C(Cc2c(C)n(C)cn2)=O)CCC(C(=O)NC2(C)CCN(C)CC2)=C(F)C1 c1(C(N2C(CNC(C3ON=C(C)C3C)=O)COCC2)=O)ncnc2c1CCCC2 Cc1ccc(O)c(C(N2CC(F)CC2CN(C)C(C2CC3CCC2CC3)=O)=O)c1 C1(N(C(c2scc(OC)c2)=O)C)CCN(C(=O)CCc2nnc(S)n2C)CC1C C1(C(=O)NC2CC(N(C(=O)CCC3CCOC3)C)C2)CCC1(F)F C(=O)(C1=CC2(CN(C(C3CCCCC(=O)N3)=O)C2)OC1)N1CCC(C)(CCC)C1 c1(C(=O)NC2(CNC(COCC)=O)CCOC2)cc2nccc(C(F)F)n2n1 C1(CC=C)(C(=O)O)CN(C(=O)NC2CCN(C(C)(C)C)C2)CCO1 C(C(C)CN(C)C(C1CCC1c1nc[nH]n1)=O)NC(COC(C)=O)=O C=CCC(C(=O)N(CCCN(C(=O)CC1CCOC1=O)C)C)NC(C)=O CCC(CCCC(=O)NC1C(C)C1C)NC(c1cc(C)cs1)=O C12(NC(CN3CC(=O)NC3=O)=O)CCN(C(c3cc(F)ccc3Cl)=O)CCC1C2 c1(OCC(N2CCCCC(NC(CCCC=C)=O)C2)=O)ccc2c(c1)OCO2 c1(CN(C(c2ccc(CNC(C3CC(COC)C3)=O)o2)=O)C)ccc(=N)[nH]c1 C1(NC(C(CC)SC)=O)CC2CC(NC(=O)C=Cc3cccc(O)c3)CC2C1 C(=O)(C(CC)C(=O)OC)N(CC(C)(C)CNC(C1CC(n2cccn2)C1)=O)CC C(C)(CCN=c1[nH]c(N2CCN3CC(C)CC3C2)nc2ccccc12)OC C(C(CC(C)C)C(=O)N(C(CC)CC)CC)NC(c1cc(CC)no1)=O C1(NC(C2CCS(=O)(=O)C2)=O)CC12CCN(C(C1CC3(C1)CC31CC1)=O)C2 c1(C(C)(C)C)nc(Cl)c(Cl)c(Cl)c1Cl.N12CCC(O)(CC1)CCC(=O)NC2=O C1(NC(c2ncc(F)cn2)=O)CC2CCCC(C1)N2C(C1CN2CCC1CC2)=O c1(C(=O)NCC2(O)CN(C(c3sccc3I)=O)C2)cc(F)c2cc[nH]c2c1 N1(C(C(C2CC(C)(C)C2)OC)=O)CC(CC(=O)NCC2(CO)CCCC2)CC1C CC1CN(C(C2(n3cnnn3)CC2)=O)CCN1C(c1coc(Br)c1)=O C1(C(=O)NCC(CC(C)C)NC(c2cc(C)nn2C)=O)CCc2ncnn2C1 c1(C(N2CC(C(N)=O)(CNC(C(C)O)=O)C2)=O)nc(C(F)(F)F)cn1C c1(C(=O)NC(C(=O)OCC)CO)cnn(-c2ccc(O)cc2)c1CC N1(C(C2C(NC(C=C(C)C)=O)CC2)=O)CCNC(=O)CC1 c1(C(=O)NCC2N(C(c3c(OC)csc3)=O)CC(O)C2)ccc2nnc(C)n2c1 C(C)(CCNC(=O)CC1CC1(C)C)N(C(C=CCOCCOC)=O)C Cc1ncc(NC(c2csc(C(F)(F)C(F)(F)F)c2)=O)c(C)c1Br c1(C(C)(F)F)cccc(C(=O)NC2CCCC(NC(C3(CCF)CCC3)=O)C2)c1 N1(C(c2ccc(OC(C)C)cn2)=O)CC(C)CCC1CNC(c1cc(O)cs1)=O c1(NC(c2cccc(-c3cnn(C4CCCCO4)c3)n2)=O)c(CO)cccc1F C1(C(N2CC(N(C(CCCCCC)=O)C)C3(C2)CC3)=O)CCc2nncn2CC1 c1(C(N(C(CNC(C(CC)n2cncn2)=O)C)CC)=O)ccc(C)nc1OC C1(CC(=O)NCC2CC2NC(=O)CC2CCOC2)CCC(C(F)(F)F)CC1 Cc1ccc(CNCC2(CN(C(=O)C=CSCc3ccco3)C)CC2)n1C Cc1cn2cc(CC(=O)NC3CN(C(=O)CCCc4cccs4)CC3F)nc2s1 C(=O)(CCCCCC#N)N1C(C=CC(N2C(C)CC2CO)=O)CCC1 C1(NC(CN(CC#C)C(C2CCCC2O)=O)=O)CC(=O)N(C2CC2)C1 C=CCCC(C(=O)Nc1ccc(F)cc1CO)NC(c1cc(C)co1)=O C12(C(=O)NCCCC(=C)C)CC(CCO1)N(C(=O)C(=O)C(C)C)C2 c1(C(C)C)ncc(Cl)c(C(=O)NCCCC(C)NC(C2CC3C=CC2C3)=O)n1 CN1CCC(C)(C(=O)NCCOCCCN(C)C(C2(F)CCCC2)=O)C1=O CC1CCc2[nH]nc(C(=O)NCC3CCCN3Cc3cc(F)ccc3F)c2C1 C1(CNC(c2c(C)nc[nH]2)=O)CC(C)N(C(=O)CCOC2CCCC2)C1 c1(C(=O)NCC(C(C)C)NC(C2OCCN(CC)C2)=O)cncn(C)c1=O c1(C(N(C(CNC(CCSCC)=O)C)CC)=O)ccc(=N)[nH]c1 C(N=c1[nH]c(=NCCCn2cnnc2C(C)(C)C)c2sccc2[nH]1)C1C(C)C1 CC1Cc2ccc(NC(=O)COC3CN(C(=O)C4CC4)C3)cc2N1 C1(C(=O)NCC2(CNC(C(C=C)(C)CC)=O)CC(F)(F)C2)CCn2nnnc2C1 N1(C(CC2C(C)=NNC2=O)=O)CCN(C(C2C3CCC(=O)C23)=O)C(C)C1 c1(C(=O)NC2C(NC(=O)CC3NC(=O)NC3=O)CC2)cnc2cccnc2c1 N1(C(C2CC3(CSC3)C2)=O)CCC2CN(C(=O)CC3CCC4CC34)C2C1 C1(O)(C(=O)NC2C(NC(c3c(C)scc3)=O)CCCC2)CN2CCC1CC2 N1(C(COc2cn(C)nc2)=O)CCCN(C(=O)C=Cc2ccncc2)CC1 c1(N(C)C)ccc2c(c1)CCCN2C(=O)C(F)(F)c1ccnn1C N1(C(c2ccc(COC(C)=O)cc2)=O)CC2(CC2)CC1CNC(C1CC(O)C1)=O C1(C(=O)NCc2ccc(C(=O)NC(C3COCCO3)C)o2)CC2(C1)CC2(F)F C1(ONC(c2ccccc2-n2cc(C3CC=CCC3)nn2)=O)C=CCC(CO)C1 C1(CNC(c2c(COC)ncs2)=O)CC(C)N(C(C2(C)COC2)=O)C1 c1(C(=O)NC2(CNC(C3C(C=C)CC3)=O)CCC2)cn(C2CC2)c(C)cc1=O c1(CN(C)C(C2CCC(F)(F)C2)=O)ccccc1CNC(C1CC(O)C1)=O c1(OCC)ccc(CNC(=O)C(=O)NCC=C2CCOCC2)cn1 Cc1ccc(NCC(=O)N(C(C)CN(C(=O)C(c2ccccc2C)C)C)C)cc1 C1(C(N(C)CC2CN(C(CC(CC=C)(C)C)=O)C2)=O)CCc2nnc(C)n2C1 S(=O)(=O)(c1cccc(C)c1)N1C(C(=O)NC(C(=O)OC)Cc2cnc[nH]2)CC1 N1(C(CSC)=O)CCC2(CC1)CN(C(=O)CC1COCC1O)C2 C(=O)(C(C(C)C)C(C)C)NC1C(NC(CN(CC)CC)=O)COC1 C1(CCC)CCCN1C(=O)C=CC(C)NC(C1(CC)CCCC1)=O C1(OCC)COCCC1CC(=O)Nc1ccc(C(=O)Nc2ccccc2)cc1 N1(C(CC(C)(C)NC(C(C)OCCC=C)=O)=O)CC2CCCCC12C c1(C(=O)NC(C)C(C)NC(c2c[nH]nc2F)=O)cccc(NCc2cncs2)c1 c12ncc(cc1Br)NC(=O)N2.c1(OC)ccc(OCCS(C)(=O)=O)cc1 C(=O)(N1CCN(C(=O)Nc2nc3c(s2)COCC3)CCO1)OC(C)(C)C CCS(=O)CC(=O)N1CCCCC1C(C)(C)CNC(=O)C=CC(F)(F)F C1(NC(C(CC)SC)=O)CCN(C(=O)CCC(=O)c2ccc(OC)cc2)C1CC Cc1cc(C)c(S(=O)(=O)N(CC(=O)NC(C)(C)C)C(C)C)cc1-c1nn[nH]n1 C12(C(N3C(C(C)(C)NC(=O)CCCn4ccnc4)CCC3)=O)CC=CC(C1)OC2 C(=O)(CCCCCCn1cc(-c2nc(C)cs2)nn1)Nc1c(SC)cccc1 CCCC(C(=O)NC1CN(C(c2onc(C)c2C)=O)CC1CC1CC1)NC(C)=O c1(OC)nn(C)cc1C(=O)NCC1CC1CNC(c1cccc(C)c1)=O c1(OCC)ccc(F)c(C(=O)N(CCNC(C2CCCN2C=O)=O)CC2CC2)c1F C1(CC)OCCC1C(=O)NCCCCN(C)C(c1cncn1C1CC1)=O C(N=c1ccc([N+](=O)[O-])c[nH]1)C1(O)CCCN(C(=O)C(C2CC2)C2CC2)C1 C1(CC(=O)NCCC(C)N(CC(=O)OC(C)(C)C)C(C)=O)CC2(CCC2)CO1 C(=O)(CCCCC(C)(C)OC)NC1CCCCN(C(CCCC#CC)=O)C1 CC1C(c2ccccc2)CCN1C(C1CCCCN1CC(F)F)=O c1(N(CCCNS(C)(=O)=O)C)nc(=NCCCS(=O)(=O)N(C)C)[nH]c2c1CCC2 C1(CNC(c2c(C)[nH]cc2)=O)CC(C)(C)CN1C(=O)Cn1ccc(C(F)F)n1 C1(OCC)COCCC1(c1nnnn1CC1CC1)Nc1cn(C)nc1O C(=O)(C(O)C(F)(F)F)N1CC(C(N(CC(C)O)CC)=O)C(C(C)C)C1 C1(CC(=O)NCC2CN(C(C)C)C2)CCCCN1C(C1(CO)CCC1)=O CCCCC(C)CCC(=O)NC(C)(CC)CCNC(c1sc(CCC)nc1C)=O CCCCCCC(CC)NC(=O)CN(C(C1C2CCC(F)(F)C12)=O)C(C)C N1(C(C(C2CCCC2)N(C)CC)=O)CCC(C(=O)N(C(C)C(=O)OC)C)C1 C(=O)(C1=CCCCC1C)N1C(C(=O)NCc2ccc(C)cc2)CSC1 Cc1cn2c(CNC(=O)CC(C(=O)O)c3ccc(Br)s3)c(C)nc2s1 C(=O)(C1=NOC(C)C1C)NC(CNC(C1(CCOC)CCCC1)=O)C(C)(C)C C(C(C)C(=O)NCC#CC(=O)NC(C1CCCCC1)(C)C)OCC CC1(C)OCCC1C(=O)NC1(C(=O)NC(C2CCC2)C2CCC2)CCSC1 c1(C(=O)NC2(C)CCC(NC(C3C(C)(C)C3(F)F)=O)CC2)noc2ccccc12 CN1CC(C(N2CCC(CCNC(c3cc(C(F)(F)F)c[nH]3)=O)C2)=O)NC1=O N1(C(C(n2ccc(C3CC3)n2)C)=O)CCC2(CC1)CC(NC(=O)C(O)C(F)(F)F)C2 c1(OCC(N2CC(NC(CCCOCC=C)=O)C2)=O)ccccc1C(F)F C1(NC(CSCC#C)=O)CCC(N(C)C(C2CCCCC2)=O)CC1 C(=O)(C(C)(CC)CC)NC(CC=C)CNC(=O)C(C)OC C1(N(C(=O)CCC2(C)CC2)CCN(C(=O)CC2(N(C)C)CCC2)C)CCCOC1 C1(CN2CCCN(C(=O)OCC)CC2)CCN(Cc2ccccc2)C2(CCC2)C1 N1(C(=O)NC(C)CN2CCOCC2)CCCC(n2cc(CCC(C)O)nn2)C1 c1(OCC)ccc2cc(COC(C3CC(C)(O)C3)=O)[nH]c2c1 Cc1ccc(=N)[nH]c1C(N1CC(NC(=O)CCOc2ccc(F)cc2)C(C)C1)=O C(=O)(C(C)(C)C(C)(F)F)NCC1CCC(NC(Cc2cn(C)nn2)=O)CC1 N1(C(CN(C)Cc2nnc(C)n2C)=O)CCC(C)C(NC(C2(C)C=CCC2)=O)C1 N1(C(C(=O)NCCC2CC2)CCC2CCCC2)CCC2(CCC2)CC1 c1(N(C2CC(=O)NC2)C(=O)CCN2C(=O)C=CC2=O)ncnc2cccc(F)c12 c1(CC)cc(N)c(C(N2CCCC(N(C(=O)CC(F)(F)C(F)F)C)C2)=O)cc1F CC1CC(C(=O)N2CC(F)(F)CC2CCNC(=O)CC2CCOCC2)=NO1 CC(CC(=O)NC1CN(C(=O)COCCc2cccs2)CC1(C)C)CC(F)(F)F C12(C(=O)NC(C(C)O)(C)C)CCCC(CCC1)C2O N1(C(CC(CC)(F)F)=O)CC(C)CN(C(c2csc(O)n2)=O)C(C)C1 C1(C(N2CCOCC2C2CC2)=O)CCCN(C2CCC2)C1.C1(C)CC1 CC1CCCC=C1C(=O)N(C1CCCN(C(=O)C=CC2CCOCC2)C1)C C1(NC(=O)CC2CC(F)(F)C2)CN(C(C2CN3CCN2CC3)=O)CC2(CCC2)C1 C(CCC(C)CC(=O)NC1CN(C(c2nn(C)cc2C)=O)CC2(CC2)C1)=C(C)C c1(C(C(C)C)C(=O)NC2CC(C)(NC(C3CC=CC3)=O)C2)ccc(C#N)cc1 Cc1ccnnc1C(=O)NC(C)(CNC(=O)C(C)Cc1cccnc1)CO c1(OC)cc(C(=O)N(C)CCNC(C2CCn3nccc3C2)=O)sc1S(N)(=O)=O c1(NC2CN(C(C3CC(C(C)C)OCC3)=O)CC2(C)C)nc(Cl)nc2sccc12 c1(SCC(=O)NC2CCN(C(CSCC(C)C)=O)C23CC3)cc(=O)n2ccsc2n1 c1(C(N(CCNC(Cn2ncc(CC)c2)=O)C)=O)cc(C)c2[nH]nnc2c1 N1(C(CCC(C)(F)F)=O)CCC(C2CCN(C(C3CCCC3O)=O)C2)CC1 C1(CNC(c2c(OC)ccs2)=O)C(C)CCN1C(c1[nH]cnc1C#N)=O C1(C2CCC2)(C(=O)NC2CC(NC(CCCOc3c(C)cccc3)=O)C2)CCC1 C1(O)(CNC(CSCC=C)=O)CC2CCC(C1)N2C(=O)CC1CCN(C)CC1 N1(C(C(C)SC(C)C)=O)CCC2(CC1)CN(C(=O)CCN1CCNC(=O)C1)C2 C1(NC(CN(C2CCC2)C)=O)(CF)CCN(C(c2nc(C(F)(F)F)cs2)=O)C1 C12(C(N(CCOCCC(=O)NC(CC=C)CO)C)=O)CCC(C1)C2(C)C C1(C(=O)NCc2ccc(OC)nc2)CC(P(C)(C)=O)CN1 O=C1NOCCC2CC=C1C2.C1(C(=O)NCCO)(CF)CC1 C1(C#N)(C(=O)NC2CN(C(c3c(C)nns3)=O)CC(O)C2)CCS(=O)(=O)CC1 c1(NC(CC2CC(NC(CC(C)(C)O)=O)C2)=O)ccc(N2CCCC2)c(C#N)c1 N1(C(CCC=CC(C)C)=O)CC(CNC(=O)C(C)CN(C)C)OC2CCCC12 N1(C(c2[nH]cc(CC)c2)=O)CCCCC(CNC(=O)Cn2ccc(C(F)F)n2)C1 Cc1nc(-c2ccco2)cc(=NCCC(C)NC(C2CC(n3ccnc3)C2)=O)[nH]1 c1(C(=O)NCCCNC(c2c[nH]c(=NC)s2)=O)cc(F)cc(Br)c1C c1(C(=O)Nc2cc(C)c(O)cn2)cc2ccc(-c3cnc4sccc4c3)cn2n1 c1(C(N2CCCC2CNC(C2(C3CC3)CC2)=O)=O)cc(Br)c(F)cc1F C(=O)(C#CC1CCCC1)N1CCC(C(C(=O)NCC(CCC)C)F)C1 N1(C(C(CC)n2ccnc2)=O)CCCC(C)(NC(c2cc(C(C)C)oc2C)=O)C1 Cc1nc(C(=O)NC2CCCC(N(C)C(c3ccncc3Br)=O)C2)cc(O)n1 C1(C(=O)NC2CC(CNC(C3CCCNC3=O)=O)C2)CCCC(F)(F)C1 c1(CNC(C(C)(C)C)=O)ccc(C(=O)NC2C(NC(=O)NC(=O)C3CC3)C2)cc1 C#CCC(C)(CC)C(=O)N1CC(C(=O)NC(C)CCC)C(F)(F)C1 N(C(=NCCCC(F)F)N1CC2CCOCC2C1)Cc1c(OC)c(Cl)ccc1 C12(SC)CC(NC(=O)Nc3ccc(N(C)C(=O)OC(C)(C)C)cc3)(CO1)C2.OC N1(C(c2ccc(C(C)=O)nn2)=O)CCCC2(CNC(C3(C)CCOCC3)=O)CC12 c1(OCCCC)ccc(N)c(C(N2CC(NC(=O)Cc3nccn3C)C2)=O)c1 N1(C(c2ccn(COC)n2)=O)CCCC(C2CC2NC(=O)C2=C(Cl)CCOC2)C1 c1(C(=O)NCCNC(C(C2CCOC2)OC)=O)cnn(CC(F)(F)F)c1C1CC1 n1(CC)ncc(C(=O)N(C2CCCN(C(=O)Cc3c[nH]nc3C)C2)CCF)c1C N1(C(C2(CC=C)CCC2)=O)C2CCCC1CC(NC(=O)C(C)(C)COC(C)C)C2 C(=O)(C1=CCCSC1)NCc1c(C(=O)NCCc2cc(C)ncc2)n[nH]c1 C1(NC(c2cc(C)sc2C)=O)CCN(C(=O)C(c2ccccc2)F)C(C)C1 c1(OC)cnncc1C(=O)NC1(CCC(=O)NCc2ncc[nH]c2=O)CCCC1 c1(C(N2C(C)CN(C(c3cncs3)=O)CC2)=O)cnn2cc(S(C)(=O)=O)cnc12 c1(C(=O)NC(C(=O)Nc2cn(C(C)C)nc2)CO)c[nH]ccc1=O c1(C(C(=O)NCC2C3CN(C(C(C#N)C4CC4)=O)C2C3)O)ccc(F)c(F)c1 CC(C)CCCCCC(=O)N1CC(C(=O)NCC23CC(F)(C2)C3)CC12CCC2 N1(C(CC(=O)NC2CC2)=O)CC2(CCN(C(=O)CC(c3cccc(F)c3)O)C2)C1 c1(C(=O)NC(C2CCCN2C(C2CCCC(=O)O2)=O)C)ccn2c1CSCC2 CC(CCCCNC(C1C2CCCC12)=O)NC(c1ccnc(OC(F)F)c1)=O c1(CC(=O)NC2C(NCc3cnn(C(F)F)c3)CCC2)cnn(CC2CCC2)c1 C1(C(=O)OC)C2CC2CN1C(=O)C(C)C(C)NC(C12CCC(OC)C1C2)=O Cn1cnc2cccc(C(=O)NC3CCC4(CC3)CN(C(C35CC3C5)=O)C4)c12 C(=O)(CC1=CCCC1)NCC1(CNC(c2c(CC)nn[nH]2)=O)CC1(F)F c1(C(=O)OCC)nc(=NCCN(C(c2cccc(Cl)c2)=O)CC)cc[nH]1 Cn1c(C(N2CCC(N(CC(C)(O)C(F)F)C(=O)OC(C)(C)C)C2)=O)cnc1Br c1(NC(C)CC(C)NC(c2ccn(O)c(=O)c2)=O)ccnc2ncnn12 CC1CCC(=CC(=O)NC(CNC(=O)C(C2CC2)N(C)C)C2CC2)CC1 C(CCN)(C(=O)NCC1CCCCN1Cc1cccc(F)c1)OC C1(NC(C2(COC)CC=CC2)=O)CC(O)CN(C(=O)Cc2ccnc(C)c2)C1 C(C(CCOC)NC(C1CC2CC2C1)=O)NC(C(F)=CCC)=O c1(C(N2C(CNC(CCc3n(CCOC)ccn3)=O)CC2)=O)nnc(O)cc1C C1(C(C)(C)NC(c2cc(C)no2)=O)CCCN(C(=O)C(CO)NC(N)=O)C1 N1(C(CNC(C(CC)CC)=O)=O)CCCCC(NC(=O)C(CC)c2cccnc2)C1 CCCC(O)CC(=O)NC(c1ccccc1)Cn1cc(-c2cnc(Br)n2C)nn1 c1(OC)cc(OC)cc(OC)c1OC.C12(CN)CCCC1C2.C1CCOCC(=O)C(=O)N1 N1(C(CCC#C)=O)CC2C(CNC(=O)C(c3ccc(OCCC(C)C)cc3)C)C2C1 c1(C(=O)NC2CCCC(NC(c3ccc(CO)o3)=O)CC2)ccn2nccc2c1 c1(OC)c(C)csc1C(=O)NC1CCCCC1CNC(C1CCC1)=O N1(C(C2(C#N)CC=CC2)=O)CCC2CC2(NC(=O)C=Cc2cccs2)CC1 C1(CCOC)(NC(=O)COCCSC)CCN(C(=O)C(C)CN2CCOCC2)C1 C1(OCC)CC2CN(C(=O)CC3(C)CCN(C(c4cn(C)nc4C)=O)C3)CC12 Cc1sc2ncc(C(N3CCCC3CNC(c3cccn3C)=O)=O)n2c1C N1(C(c2cccc(OC)c2F)=O)CCC2(C1)CN(C(=O)C(C)=O)CCO2 CCCCC(O)CC(=O)N1CCCC1C=CC(=O)N(C1CCN(C)C1)C CCC(C)C(=O)NCC(=O)NCC1(C)CC(NC(=O)Cc2cc(C)on2)C1 C1(NC(C(F)=CCC)=O)CCCC12CCN(C(=O)C=CCCC)CC2 CC1CN(C(C2CNC(=O)N2C)=O)CC1NC(=O)Cc1cnn(C)n1 c1(CC(=O)NC2CC3CCC2(NC(=O)CCCN2CC2)C3)c[nH]c2ncccc12 c1(CNCCN2C(NC(=O)OC(C)C)CCCC2)cc(Cl)c(F)c(Cl)c1 N1(C(C(C)O)=O)CC(CO)C2(C1)CN(C(c1cc(P(C)(C)=O)ccn1)=O)C2 N1(C(c2cc(C(C)=O)on2)=O)CC(NC(c2ccc(OC(C)C)nn2)=O)C(C)C1 CC(C)CC(C)(O)C(=O)N1CC2CCCC2(C(N2CCCC(C)(F)C2)=O)C1 C1(C(N2CCCC(C(=O)OC)C2)=O)CCCN1N1CCN(C(C)=O)CC1 N=c1[nH]c2c(C(=O)NCCCCNC(C3CC(n4cnnc4)C3)=O)cccc2o1 C=CC(C)(C)CC(=O)N1CC(OC)CC(NC(=O)C(N2CCC(C)CC2)=O)C1 C1(C(C)C)CN(C(=O)C(C)C(C)O)CCN1C(=O)C(F)CC1CCOC1 c1(C(N2CC(CNC(c3cccs3)=O)C3C2C3)=O)cccc(O)c1Br C1(C(=O)NC(c2ncc(C)s2)C)CCCCC1NC(=O)C(C)Oc1ccccc1 N1(C(C=CCC)=O)CCC(N(C(=O)C2=CCCC2)CC)CC1 N1(C(CCSCC)=O)CCN(C(c2ocnc2C)=O)C(C)C1C c1(C(N)=O)cnc(NC(c2nc(CNC(=O)CC3CC34CC4)cs2)=O)c(Cl)c1 C(=O)(C1=C(Cl)CCC1)NC(C(=O)NCCCN(C)C)C1(C)CC1 C1(O)(C(CNC(C2C(OCC)C2C)=O)(C)C)CN(C(=O)C(n2ccc(C)n2)C)C1 C(CC(C(C)C)NC(=O)CC1CC(C)=NO1)NC(CCNS(CC)(=O)=O)=O c1(C(=O)NCCC2CCN(C(C3CC4CCC(C3)O4)=O)C2)c(F)ccc(Cl)c1F c1(SC)cc(C(=O)NCC2CCN(C(C3CCCCO3)=O)C2(C)C)ccc1N C1(C(=O)NC2(C(=O)NCCOCCOC)CCSC2)CC2COCC2C1 C(=O)(C(C)(C)CCCNC(c1ccccc1C#N)=O)NC(C(C)C)CN(C)C c1(C(=O)NCC(CN(C(=O)CCCNC(C)=O)CC)(C)C)cc2cscc2s1 C#Cc1cncc(C(N2CCC(OCC(=O)Nc3ccc(C(C)C)cc3)C2)=O)c1 C1(NC(C2C(=C)CC2)=O)CC(C2CCN(C(c3ccc4nnn(C)c4c3)=O)C2)C1 c1(C(N2CCC(N(C(=O)CCCCCSC)CC)C2)=O)ccc2sncc2c1 c1(C(N(CCNC(CCn2ccc(C)n2)=O)C(C)C)=O)ccc2c(n1)CCCC2 CCCCC(CN(C(=O)C(CC1CC1)NC(=O)Cn1c(O)nnc1O)C)CC c1(C(N(C2CN(C(C(C)NC(N)=O)=O)C2)C)=O)cccc2c1C(=O)NC2=O C#CC1(N(C)C)CN(C(=O)C(C2CC=CCC2)NC(c2nocc2Cl)=O)C1 C#CCC(C)(CC)C(=O)NCc1cc(C)c(C(=O)N(C)Cc2ccccn2)o1 C1(C)(CNC(CCOCC#C)=O)CCCN1C(C1COCCOC1)=O Cc1cc(C(N)C(=O)NC2(c3ccncc3)CCC2)cs1 N1(C(CC2N(C(CCOCC(C)C)=O)CCC2(C)C)=O)CCOC2COCC12 c1(C(=O)OC)cnc(CNc2ncc(Br)c(Br)n2)c(F)c1 C(CN=C(NC1CCC1)N1CCc2nc(O)nc(O)c2C1)c1cc(C)c(C)cc1 c1(C(=O)NCC(CO)NC(C2OCC(C)(C)C2)=O)cc(Cl)c(Cl)cc1N CC1CN(C(c2cnnc(-c3ccccc3)c2)=O)CCN1C(C1(F)CCOC1)=O C#Cc1ccccc1NCC(=O)Nc1cccnc1OC CCC(C)C(C(=O)NC1CCCN(CC)C1)N(C(=O)C(C)n1cnnn1)C C1(NC(COCCC#C)=O)CCN(C(=O)C(c2ccc(F)cc2)(C)C)CC1CO c1(C(=O)NC(C2(O)CCN(C(=O)CN3CCCC3)C2)C)nc2c(s1)COCC2 N1(C(N)=O)CCOC(CCNC(=O)C=CC(=O)NCCO)C1.C1(N)CCS(=O)(=O)C1 O=C1CCCCC(C(=O)NC2(C(=O)NCC3CC(C4CC4)=NO3)CCC2)N1 N(C1c2ccccc2CC1NC(C1C(C)C1(F)F)=O)C(C(CC)n1cncn1)=O c1(NC(CC(C2CC2)NC(CC(CC)(F)F)=O)=O)ccc2occc2c1 N1(C(=O)OC(C)(C)C)CCC2(CC1)CC(C(=O)NCC1(c3cccs3)CC1)CO2 CC1CCN(C(C2CCCN2N=O)=O)CC1N(C(=O)CCc1ccc(Cl)cc1)C N1(C(CNC(=O)OCC)=O)CCCCC(NC(=O)CCC2(C)CC2)C1 Cc1cn2c(n1)CC(C(=O)NC(C)CNC(C1(CCN(C)C)CC1)=O)CC2 N1(C(c2ccn(C)c2)=O)CCN(C(=O)CCc2cccn2C)C2CC12 c1(C(C(=O)O)NC(C2CCC3(CC2)CC3)CC)ccc(OC)c(OC)c1C c1(CC(N2CC(O)(CNC(C(C)C3CCCO3)=O)C2)=O)ccc2n[nH]cc2c1 C(C)(C1OCCc2ccccc21)NC(=NCc1cc(C)cc(C)c1)NCC1CC1 C1(C(=O)NCCC2(O)CN(C(C(C)c3ccon3)=O)C2)CCc2ccccc2C1 O=C1CCC(NC(=O)CN2CCN(C(C34CSCC3C4)=O)CC2)C(=O)N1 C1(C)(NC(C(COC)NC(c2ccsc2C)=O)=O)CCC(=O)NC1=O N1(C(C=C(C)C)=O)CCC(CO)C(NC(=O)CCCCN(c2ccccc2)C)C1 C(=O)(CCCCC#N)N1CC(C)C(NC(C2CCCCN2C)=O)C1 c1(NC(Cc2nc(C)on2)=O)ccc2c(c1)NC(=O)CCC2.N12C(CC3CC13)C2=O C(=O)(C1CSc2ccccc21)N1CC(C)C(CNC(=O)CCC2CC2(F)F)C1 C(C)(C)(CCC(=O)NC1CCC(NC(=O)CCc2ncc(C)[nH]2)CC1)OC C1(NC(C2CC(O)(CC#C)C2)=O)CCC(C)N(C(c2cccc(OC)c2N)=O)C1 C1(NC(C(COc2ccccc2)OC)=O)CCC12CCN(C(=O)C(F)F)CC2 C(=O)(CS(=O)(=O)c1ccccc1Cl)NC1C(NC(Cn2ccc(C)n2)=O)CCC1 C1(C(F)(F)F)(OC)CN(C(=O)C=Cc2ccncc2)CCO1 CCC(CC1CCCC1)C(=O)NC1CCCC1CNC(=O)CC(F)(F)F Cc1nc2cccc(C(=O)NC3CC4CCC3CN(C(=O)C=C3CCC3)C4)c2[nH]1 Cc1cccc(C(=O)NC2CCCN(C(c3coc(-c4cccnc4)n3)=O)C2)n1 c1(OC)ccc(CNC(=O)C(C)CNC(C23CC(C#N)(C2)C3)=O)cc1 c1(OC)cc(CNC2CCN(C(c3ccnnc3)=O)C2)cc(CC2CC2)c1O C1(NC(c2c(OC)ccs2)=O)COCCN(C(c2cccc(=S)n2O)=O)C1 C1(C(=O)NCC(C2CC2)NC(C2CC3(CCC3)C2)=O)CC2(CCCCC2)C1 S(=O)(=O)(c1cccc(Cl)c1Cl)N1C(C(=O)Nc2cnn(CCO)c2)CC1 C#Cc1ccnc(C(=O)NC2CCCC2NC(c2nc(Br)c[nH]2)=O)c1 c1(CC(C)C)cn(CCNC(=O)CC2CCOC2C(=O)O)nn1 CCCCC(O)C(=O)NC1CCCC1NC(c1cnn(C(C)C)c1F)=O N1(C(C2CCC(CCC=C)C2)=O)CCC(c2ccc(CO)cc2)CC1 N1(C(c2c(C)nn(C3CC3)c2)=O)CC2(CC2)CC1CNC(=O)CC1C=CCCC1 c1(C(=O)NC(C(=O)NC2C(C)CN(C)C2)C(C)(C)O)c[nH]c2nccc-2c1 C(=O)(C1CSc2ccccc21)NC12C(C)OC(CNC(c3c[nH]c(=N)s3)=O)(C1)C2 Cc1cc(N)c(C(=O)NC2CS(=O)(=O)CC2N2CCCC2)nc1C c1(C(N2CC(OCC(N3CCC(OCC(N)=O)C3)=O)C2)=O)ccc(O)cn1 N1(c2c(C(C)=O)cnc(Cl)n2)CC(NC(=O)C2=COCCO2)CC2(CC2)C1 C1(NC(=O)OC(C)(C)C)CCCCC1c1nc(-c2cccnc2S)no1 C(=O)(C1=NOC2(CCC2)C1)NCC(CCC)C(=O)NCCCc1cc(C)no1 S(=O)(=O)(c1cccc(-c2cccc(C(=O)N(C)CCC3CCCN3C)n2)c1)NC C1(NC(c2cc(C)oc2)=O)CN(C(C2CC2c2ccc(Cl)cc2)=O)CCC1(C)C C12(CNC(c3cc(CC)oc3C)=O)CCC1CCN2C(=O)CCCN(C)C n1(CC(=O)NC2CC(c3cccc(Cl)c3)C2)c(-c2cccnc2)noc1=O c1(OC)ccc(COC(C2C(C)CN2C(=O)OC(C)(C)C)=O)cc1 C(CCCCC(=O)NCCCC(C)(C)C)N(C(c1cnc(CC)nc1)=O)C C1(NC(C2CC(O)(CNC(=O)CSC(F)F)C2)=O)CCC(C2CC2)C1 c1(CNC(C(CCCC)C)=O)cnn2c1CN(C(=O)CCCc1cnn[nH]1)CC2 CC1CC(NC(=O)COCCO)CCN1C(c1nnn(C)c1N)=O c1(C(=O)NCCN(C)C(c2cnc(C(F)(F)F)nc2)=O)cc(Cl)c(F)cc1O C#CC1C(C(N2CCCC(N(C(=O)CCc3ccc(Cl)cc3)CC)C2)=O)C1(C)C c1(CNC2C(C(=O)NCc3ccc(-n4cnnc4)cc3)C2)cc(Cl)c(O)c(Cl)c1 c1(C(=O)NC2C(NC(C3(C#C)CCCC3)=O)CCOC2)cccc(S(C)(=O)=O)c1 c1(OC)cccc(CN2CCC(SC)C2)c1OC(c1ccccc1)C C1(N(C(C2C(C#C)C2)=O)C)CCCN(C(c2ccn(-c3cccc(F)c3)n2)=O)C1 C1(C(NNC(=O)C2C(C)OCC2)=O)CCC(C#N)(N)C1.C(=O)O C12(NC(CCCC=C)=O)CCC(CC1NC(c1cccc(-c3nnco3)c1)=O)C2 Cn1c(C(=O)NC2CCCC2CNC(=O)C(=Cc2c[nH]cn2)F)ccc1[N+](=O)[O-] c1(C(=O)NCc2c(C(NOCC(CC)C)=O)[nH]cc2)cc(C)ccc1C C(=O)(C1COc2c(F)cccc21)NCc1c(OC)cc(Br)c(C)c1 C(=O)(CCC(C)C#N)NCCCCCNC(CSCC#C)=O c1(C(=O)NC)ccc(S(=O)(=O)N(c2ncncc2I)C2C3CNCC23)cc1 N1(C(c2c(C)cc(SC)s2)=O)CCC2CCN(C(=O)C=CC(C)(C)SC)CC12 c1(C(=O)NCC(CO)NC(C2CC(F)(F)C2)=O)ccc(=NCC2CC2)[nH]c1 c1(N2CCCC(C(=O)NC(C(=O)OC(C)C)C)C2)ccnc2cc(Cl)ccc12 c1(CC)c(C(=O)NCC2CCC2NC(c2ccc[nH]2)=O)nnn1-c1ccccc1 C1(C2CC2)(NC(C2N(C(c3cc(C)c(N)cn3)=O)CC2)=O)CCCCC1 N(C1CCn2ccnc21)C(N(C)CC1OCCN(C)C1)=O N1(C(C=CC)=O)CCC2(CC1)C(NC(=O)C=Cc1cc(Cl)ccc1Cl)CS2(=O)=O CC(C)(CCCNC(c1ccc(C#N)cc1)=O)C(=O)NC(c1cscn1)CO N1(C(CC)=O)CCN(C(=O)CCOc2ccc(OC)cc2)CC1CC C(=O)(C(CCC=C)NC(C1CCCC(=O)C1)=O)NC(CC#C)C(=O)OC c1(OC)cc(F)ccc1NC(C1(CNC(=O)Cc2csnn2)CCCC1)=O CC1CN(C(=O)CN2CCCC2=O)CC2(CCN(C(C3CCCSC3)=O)C2)O1 CCC(CC)C(F)C(=O)NCC1(C)CCCN1C(=O)CCCn1cncn1 C1(CNC(C2(C)CCN(C(C)=O)C2)=O)C(C)CCCN1C(c1cccc(C)c1)=O c1(NC(c2n(CCC)ccn2)c2nnnn2CCSC)cc(F)c(Br)c(F)c1 c1(OC)ccccc1C=CC(=O)NC1CCN(C(=O)Cn2ncc(Cl)c2C)C1 c1(NC(=O)NCC2CC(N(C)C)C2)nc2nccc(=O)n2[nH]1 c1(C(=O)NCCN(C(c2cc(C3CCOCC3)no2)=O)CC)cnc(C)cc1Cl N1(C(C(CC#N)c2ccccn2)=O)CC2CCC(C2)C1 Cc1cc(NC(CNC(c2ccc(CC(C)C)cc2)=O)C2CC2)ccc1[N+](=O)[O-] c1(N2CCC(N(C)C(c3ccccc3C(=O)NCCF)=O)C2)ncnc(Cl)c1F N1(C(C(COC)OC)=O)CCOCC(NC(C2(C)CCCC2C)=O)C1 CCCCC(C(=O)NCCNC(c1c(C)cc(O)nc1C)=O)C(C)C C1(C(=O)NCC2(F)CCN(C(=O)C(F)C3CCC3)CC2)CC2(CCCC2)CO1 CCCC(C(=O)NCC1CCCC(Cn2cc(CSC)nn2)C1)C(=O)O c1(CC(C(=O)OC)OC(=O)C(C)c2ccco2)ccc(F)cc1 C1(CC(=O)NC(CC)(C)CN(C)C)CC(C)(C)CO1.C1(=O)C(C)CN1 C1(C(N2CCC(CNC(CC)=O)C(O)C2)=O)CN2CCCCC2CO1 N1(C(C=CCOC)=O)CCN(C(=O)CC2CCCC(=O)C2)C(C)C1C c1(OC)nc(C)ncc1C(=O)NC(CNC(=O)Cc1n[nH]c(C)n1)C1CCC1 N1(C(C2(CNC(C3(C#N)CC3)=O)CCCC2)=O)CCC(O)C(F)C1 c1(C(=O)NCC(C)CNC(C2CC2C2CCCCC2)=O)ccc(N=S(C)(C)=O)s1 C(=O)(CCC(F)(F)C(F)F)NC1CN(C(COC(CC)C)=O)CC(O)C1 C1(CNC(COC2CN(C(C(C)SC)=O)C2)=O)CCCC(N(C)C)C1 C1(NC(C2C(=C)C2)=O)(CO)CCCN(C(C2CC(O)(C#N)C2)=O)C1 c1(SC)ccc(N)cc1C(=O)NC1COCCC1NC(C1CCC(=O)NC1)=O N1(C(COC(CC)(C)C)=O)CCCC(C(C)(O)CNC(=O)C#CC(=O)N(C)C)C1 C1(CCC(N2C(CC(=O)NCC(C)(C)OCCO)CC2)=O)CCCCC1 N1(C(c2ccc(NC(C)=O)nc2)C(=O)NCC2CCCO2)CC2COCC2(C)C1 C(=O)(C(CC(F)F)NC(=O)CC1CC2(CC2)C1)N1C(C(=O)OC)C=CC1 C1(C(=O)NC2(C3N(C(C4N(C)CCC4)=O)CCC3)CC2)CCC2CC2C1 C#Cc1ccc(F)cc1C(=O)NC1CCCC12CN(C(=O)C(C)OC)C2 C1(C)(CNC(CCC(C)O)=O)CCN(C(C2CC2C2CCCC2)=O)CC1 N1(C(CCNC(=O)NC)=O)CC2(C)CN(C(C3(C#N)CCSCC3)=O)CC2(C)C1 C(=O)(C(C(C)NC(c1ccc(C2CC2)o1)=O)C(C)C)NCc1c(C)scc1 C(=O)(CCC(C)CN(C)C)NCC1C(NC(c2nncc(OC)c2)=O)C1 N1(C(CCOCCCOC)=O)CC(NC(C2CC2[N+](=O)[O-])=O)C(C)C1 c1(CC(=O)NCC2CC2NC(c2nocc2Cl)=O)cc(F)cc([N+](=O)[O-])c1 c1(NC(C(CC)C)=O)cc(C(N2CCC(C(=O)NC)CC2)=O)n(C)c1 CCC(CC(F)F)C(=O)N(CCCOCCN(C(=O)Cc1ncoc1C)C)C c1(C(=O)NCC(CO)NC(=O)Cc2ccc(SC3CC3)cc2)cn2c(n1)SCC2 CCC(CC(=O)N1CCCC1CN(C(=O)CCc1ccc[nH]1)C)C(C)(C)C c1(C(=O)NCCN(C(C(C)NC(N)=O)=O)C)cc(O)cc(F)c1 c1(C(N2CCCCC(N(C(=O)C(CO)N(C)C)C)C2)=O)ccc(N=[N+]=[N-])cn1 C1(C2CCN(C(c3cc4c(F)cccc4[nH]3)=O)CC2)(NC(=O)CC=C(Cl)Cl)CC1 Cn1ccc(C(=O)NC23CCC(NC(C4CCOC(C)(C)C4)=O)(C2)C3)cc1=O c1(C(N(C2CN(C(C3(C=C)CCC3)=O)CC2F)C)=O)cc(Cl)c(OC)c(Cl)n1 c1(NCC2CCCCN(C(C(C)=C(C)C)=O)C2)cc(=O)n(C)c(O)n1 C1(NC(CC)=O)CN(C(=O)C=Cc2ccccc2F)CC2(CCC2)C1 Cc1[nH]nc2ccc(NCC3(C)CCNC3)nc12 c1(C(N2CC(C)(CC(=O)Nc3ncccc3Cl)C2)=O)cc(CO)cc(Br)c1 N1(C(COCC(C)(C)C)=O)CCCC2C(NC(c3c[nH]ccc3=O)=O)C(C)(C)C12 c1(C(N2CCC(C)(CNC(C3CC3C#N)=O)C2)=O)c(OC(F)(F)F)cccc1F c1(C(N2C(c3cn(C)nc3)CCC2)=O)cccc(NC(=O)NC(C)(C)C)c1 C1(C(N2CC(C)(OCC(=O)NCC(C)(C)C#N)C2)=O)CC1C1CCCC1 c1(C(N2CC(CNC(CCOCC)=O)C(C)C2)=O)nn(C)cc1S(C)(=O)=O C12(C(=O)NCC3CCN(C(COCCCC)=O)C3)CCC(O)C1CC2 N1(C(C2CN(C(CNC(C=C)=O)=O)C2)=O)CCc2nn(-c3ccccc3)cc2C1 C(=O)(N1CC(C)(O)CO1)C1CCN(C(c2cc(C)c(O)nn2)=O)C1C C1(C(N2CCC(CNC(COCCC)=O)C2)=O)CCOC(C)(CC)C1 S(=O)(=O)(c1cccs1)C(=O)NCCCOCCNC(C1(C2CC2)CCC1)=O Cc1c(C(=O)NC(C)(C)CNC(c2cc(F)c(F)c(F)c2)=O)cc(O)cc1N C1(C#N)(C(=O)NC(C2(CNC(=O)Cc3c[nH]ccc3=O)CC2)C)CC2CC2C1 C1(C(=O)NC(CC)C(=O)NC2CCCN(CC)C2)Cc2nccn2C1 C1(C(=O)NC(C(CO)NC(C(C)OCCN(C)C)=O)C)CC2C=CC1C21CC1 C1(NC(=O)C(F)CC2CC2)CC(N=c2nc(CC3CC3)[nH]s2)C1 N1(C(CC(=C=C)C)=O)CCCC1C1CCCN1C(=O)C=NOC N1(CC2(CN(C)Cc3cccc(CO)c3)CC2)CCC(F)C(C2CCCO2)C1 c1(C(N2CC(NC(CCC)=O)C(C3CC3)C2)=O)cccc(OC(C)C)c1[N+](=O)[O-] C1(CNC(=O)CCCCCF)CC2(CO1)CN(C(c1cccc3ccsc13)=O)C2 Cc1[nH]nc2ncc(C(=O)NCCNC(=O)CC3CCOC3)cc12 CC(C)(C)CCCCCC(=O)N1C2CCC1CC(F)(CNC(c1ccns1)=O)C2 c1(OC)cnc(F)cc1C(=O)NC(C)CC(C)NC(C1(CO)CCC1)=O CS(=O)(=O)c1cscc1C(N1CC(F)(CNC(c2cc3n(c2)CCOC3)=O)C1)=O c1(CC)nnc(C(=O)NCC2CCC(NC(=O)C=CSC)C2)s1 N1(C(Cc2c(C)noc2C)=O)CC2CC(NC(=O)C(C)(C)C(C)C)C1C2 C1(CNC(C2C=CCC2)=O)CN(C(=O)C(=O)C(F)(F)F)CCC12CCOCC2 C(=O)(C(CN(C)C)N(C)C)NCCOCCNC(C=C(CC)C)=O Cc1cnncc1C(=O)NCC1(CCNC(=O)C=Cc2scnc2C)CC1 N1(C(c2ccc[nH]2)=O)CCCC(C(N2CCCCC2CO)=O)C1 C1(CNC(Cn2nnc(C)n2)=O)CCCN(C(C2CCCN(C(N)=O)C2)=O)C1 C#Cc1cnc(N(C)Cc2cccc(C)n2)c(C)c1 c1(OC)ccc(-c2nc(CC(N3CCCC3Cc3ccco3)=O)cs2)cc1OC c1(CC)cc(C(=O)NC2CC(CNC(c3cnnc(O)c3)=O)C(O)C2)c(C)nn1 Cn1cccc1C(=O)NCCC1CC(NC(C2CC(C)(C(C)(C)C)C2)=O)C1 C1(CC)CN(C(c2ccc(Cl)s2)=O)CCN1C(=O)CC(C)OC c1(-n2c(CSCC(C)C)nc(-c3cccc(Cl)c3)n2)cc(Cl)nc2ncccc12 CCCCC(F)C(=O)N1CC2C(CC(=O)NCC3CC(C(C)(C)C)C3)C2C1 C1(NC(c2ccc(OC)nc2)=O)CCC(C)N(C(=O)Cc2c(C)cccc2C)C1 CC1(C)CC=C(C(=O)NCC2(NC(=O)Cc3cc(Cl)sc3Cl)CC2)CC1 C1(C(N2CCC(OCCNC(CC(=C)C)=O)C2)=O)CCCCC(F)(F)C1 C1(C(=O)NC(c2c(C)ncs2)C)CN(C(C2CCC2(F)F)=O)CC12CCC2 C1(C(=O)NCC2(O)CC(NC(C(C)(C)OC(C)C)=O)C2)CCC([N+](=O)[O-])CC1 C(=O)(C1=CCOC1)N(C)CCNC(C1CCN(c2nc(=N)[nH][nH]2)C1)=O c1(C(N(C(C)CNC(C23CC(C)C2C3)=O)CC)=O)cn(CC(N)=O)nn1 N1(CC(=O)NCC(CNC(C2(COC)CCC2)=O)F)CCOCC1 c1(CC)nnc2n1CCCC2C(=O)NCC1CCN1C(c1ccc(C(N)=O)s1)=O c1(SC(C)C(=O)NCC2CN(C(=O)CC3CCCC3(F)F)C2)ccccc1Cl C(N=c1nc(-c2ccsc2)c(F)c[nH]1)C1CCN(C(C(C(CC)C)C)=O)CC1C c1(CCC(=O)OC)cccc(C(O)C(=O)NCCOC(=N)O)c1 Cc1nn(CC(=O)NC2CCC(C)N(C(=O)C3=NNC(=O)C3)C2)c(C)c1Br C1(CNC(c2nncs2)=O)CN(C(=O)CC2CCCS(=O)(=O)C2)CCCO1 C#Cc1cccc(C(N2CCC(CN(C(c3ccc(C(N)=O)[nH]3)=O)CC)C2)=O)c1 CC(CCC(=O)N1CCN(C2CCCN(C(=O)CSc3nc[nH]n3)C2)CC1)N(C)C c1(CC)nccn1CCC(N1CCC(C(C)NC(=O)CN2CC(C)(OC)C2)C1)=O C(=O)(C1=CCCOCC1)N(CCCCCNC(c1cccnn1)=O)C Cc1ncc(C(=O)NCCCC2(NC(C3CC(C)CCO3)=O)CC2)c(C)n1 C1(NC(C2C(OC)CCC2)=O)CCN(C(C2CN3CCN2CC3)=O)CC1F c12ncccc1C(=O)N1CC(C1)Cc1cn(nn1)C2C.C1(OC)CC(C)(CC)C1 CC(C)C(CCNC(=O)C(C)CSC(F)(F)F)NC(=O)CC1CCCO1 c1(OC)ccc2c(C)c(C(=O)NCCC(O)CNC(c3cnc(Cl)s3)=O)[nH]c2c1 S(=O)(=O)(c1cccnc1NCC1C(F)(F)C12CCC2)NC1CN(C)CCN(C)C1 c1(C(=O)NC(C2CN(C(C(CC)(C)CC)=O)C2)C)c(F)ccc(OC(F)F)c1F N12CCCCC1CC(C)C(NC)=CN=NC=CC(=O)NOCC2=O C1(NC(=O)NC(C(=O)OC)C)CN(C(C2CCN(C(C)C)CC2)=O)CCC1F N#CC1(C(=O)NCC=CCNC(c2ccc(-c3cccnc3)cc2)=O)CCCOC1 C1(N(C)C(C2CC2F)=O)CCC(NC(c2cnc(C(N)=O)cn2)=O)CC1 C1(NC(c2c(C)ocn2)=O)CCCCC12CCN(C(C1CCC(C)C1)=O)CC2 N(C(=NCCCCl)NCCOC1(F)CCCN(C(C)(C)C)C1)CC(C)(C)C C(CCC1CC1)(C(=O)NOCC1CCCO1)N(C(=O)CC(=O)NC1CC1)C CC1CCC(NC(=O)C(F)(F)c2nccn2C)CN1C(C1CCOCC1)=O N1(C(C2CC23CCN(Cc2cccnc2F)C3)=O)CCC2(CC1)OCCO2 C1(C(C(=O)NC2CC(F)(CNC(C(COC)C)=O)C2)C)CCC(C)(C)CC1 C1(C)(OC)CCN(C(=O)C(=O)N(C)CC2CC(C)(C)C2)C1 C(=O)(C(C1CCCO1)C1CN(C(C(C)Cc2ccsc2)=O)C1)OC.C1(=O)C(C)O1 c1(OCC)ccc(C(=O)NC2CNC(C)(C)C2)cc1[N+](=O)[O-] C1(CN(C(COCCC)=O)CC)CCCCN1C(c1ocnc1C1CC1)=O C1(C(=O)OC)CCCC(NC(N(c2c(C)cccc2C)C)=O)CC1 CC1COCC(C(N2CCOCC2CC(N2CC(S(C)=O)C2)=O)=O)O1 C1(CNC(C(C#C)(C)C)=O)CN(C(c2cnc3[nH]cncc2-3)=O)CCC12CCC2 CC(Cn1cccn1)CN=C(NCCC1CCOC1)N(C)CCc1ccccc1 Cc1ncc(C(N2CCCC2C2(C(=O)NCCC(C)(C)F)CC2)=O)cn1 C1(NC(C=CCC)=O)CCN(C)C12CCCN(C(c1ncc(F)cc1F)=O)C2 C(=O)(CCCC(=O)N(CCCNC(C1(C)CC(C(F)(F)F)C1)=O)C)NC(C)C C(CCCC(=O)NC1CCN(c2cccnn2)CC1)(OC)OC c1(C(N2CCC(N(C(C3=NOC(C)C3)=O)C)CC2)=O)cc2nc[nH]c2cc1F C1(C(=O)NCC2N(C(CN(C(=O)OC)C)=O)CCC2)CC2CCC1C2 C#Cc1ccc(C(=O)NC(CNC(C2C3CC4C(C3)C24)=O)CC(C)C)c(C)c1 CCCCC(O)CC(=O)N1CCC(C(=O)NCC(C)S(C)(=O)=O)CC1(C)C CCCCCC(C(=O)N1CCOCC1c1ncnn1CC)=Cc1ccccc1 CCC(O)(CC)CCNC(=O)CC1(C)CCOCC1 C1(c2cn(C3CCCN(C(c4cccnc4O)=O)C3)nn2)(OC)CCCCC1 Nc1cc2c(cc1-c1ccc(NC(c3cccc(F)c3)=O)cc1)OCCO2 C(=O)(C1CCCc2cncn21)N1CC(NC(=O)CNc2ccccc2Cl)C1 CCC(CNC(=O)C(CC)C(F)(F)F)(CC)C(=O)NC1CCN(C(C)=O)CC1 c1(CCNC(CCN(CCC)C)=O)ocnc1CNC(=O)C(CC)SC Nc1cc([N+](=O)[O-])ccc1C(N1CC2CC(NC(C3CCC(F)(F)C3)=O)C1C2)=O c1(OC)cc(C(N2CCN(CCn3cc(C)cn3)CC2)=O)ccn1.C12CN(C1)C2 CC(C)CCC(=O)NC1CC(NC(C2(Cc3cnn[nH]3)CCOCC2)=O)CC1O C1(CNC(C(CC)=CCCC)=O)CCC(C)(C)CN1C(c1ncccc1N)=O C1(CNC(C(C)(C)C#N)=O)COCCN(C(=O)C=Cc2ccc(C(F)F)cc2)C1 C1(NC(CCc2cc(C)on2)=O)CN(C(c2cc3c(s2)CCC3)=O)C2(CCC2)C1 c1(C(CC(=O)NCCN(C(=O)C(F)(F)c2cccnc2)CC)C)ccc(C)cc1 CCC(F)(F)C(C)(C)C(=O)NC1CC2(CCN(C(C3(O)CCC3)=O)C2)C1 N(C1CCCOc2ccccc21)OC(CN1CCC(C2CC(C(C)(C)C)C2)C1)=O n1(CCCC)nccc1C(N1CC(CO)(NC(C2CC2C)=O)C1)=O N1(C(c2ccc(CC)cc2N)=O)CC2CCN(C(=O)C(N3CCOCC3)C)C2C1 c1(NC(C(CC)C)CO)ccc(C(F)(F)F)cc1S(=O)(=O)NCCn1cccn1 c1(OC)ncnc(C(N2CC(NC(=O)CCn3c(C)ccc3C)C(C)C2)=O)c1F c1(C(CNC(c2cc(CO)on2)=O)NC(C(C)O)=O)ccc2ccccc2c1 C1(C(=O)NC(C(C)NC(=O)CC2(C)CCOCC2)CO)CCCS(=O)(=O)C1 c1(CC)onc(C)c1C(=O)NC1CC(n2cc(C3CC(F)(F)C3)nn2)C1 N1(C(C(CC2N(C(C=CC(CC)C)=O)CC2)F)=O)CC(C(=O)NC)CC(C)C1 C1(NC(c2c(CC)scc2)=O)CC2CCC1(C(=O)NCc1ncc(Cl)cn1)C2 C=C(Cl)CC(C(=O)NCCOCCC)NC(c1ccsc1Cl)=O C1(CNC(=O)Cc2ncc[nH]2)CCC2CN(C(C3CCOC3)=O)CC12 N1(C(c2cc(F)cc(I)c2)=O)CCC2C1CCN2C(c1ccc2scnc2c1)=O Cc1cn(C)nc1C(=O)NC1CC(O)C1CC(=O)NCc1nnc(O)o1 C12(NC(c3oc(C)c(CO)c3)=O)CCCC1CN(C(=O)CN1CCS(=O)CC1)C2 CCCCC(CNC(C1(C(C)C)CC1)=O)NC(=O)C(F)CC N1(C(c2nc(C)nc(O)c2)=O)CCC(F)(F)C(CNC(=O)CCC2CC2(F)F)C1 c1(C(=O)NCC(N(C)C(C2(C(=O)NC)CCC2)=O)C2CC2)cccc(F)n1 c1(C(N2CCC(CNC(=O)C(F)(F)C(F)F)C23CCC3)=O)cc(Cl)c(F)c(Cl)c1 C1(NC(=O)COC(F)F)CCN(C(=O)C(c2cc(F)cc(Cl)c2)=O)CC1O c1(NC(C(C)OC(c2ccc(CC)cn2)=O)=O)cc(F)ccc1OC c1(CC(=O)N(C2CCN(C(=O)CSC)C2)CC)ccc(F)c(OC)c1 c1(C(=O)NC2C(NC(C(CN(C)C)(C)N(C)C)=O)CCCC2)cccc2nn[nH]c12 c1(C(N2CC(CC)OCCC2)C(=O)NCCC#N)cc(F)cc2c1CCC2 C1(CNC(=O)C(N2CCC(C3CC3)C2)=O)Cc2ccccc2CO1 N1(C(COCC(=O)NC)=O)CC(CNC(=O)CC(C)C(=O)OC)C2(CC2)C1 C#CC1CCC(NC(=O)C(=O)NCCc2cn(C)nn2)C1 C1(NC(N=c2[nH]cc(CC)nc2)=O)CCC2(CCCCC2)C1 c1(OC)c(F)c(C(N2CCC(NC(c3cnc(C)cn3)=O)CC2)=O)cc(F)c1F N1(C(c2cc(CC)no2)=O)CCC2CCCC(C1)N2C(=O)CCC(C)N(C)C C(=O)(C1Cc2ccccc21)N(C(C)CNC(c1cnns1)=O)C c1(NCC2CN(S(C)(=O)=O)C2)ccc2ccc(Cl)c(Cl)c2n1 c1(N(C)C)ncc(C(=O)NCC2(F)CC(NC(C3(C)CCCO3)=O)C2)o1 C=CC1CN(C(c2cncc(C3CC3)c2)=O)CC1NC(C1CC(CC)C1)=O C1(NC(Cc2cccc(C(N)=O)c2)=O)CCCC12CN(C(=O)CN1CC=CC1)C2 COn1cnc(C)c1C(=O)NCC(O)CC(=O)NC1COCCOC1 C(C)(CCCCNC(c1sc(N(C)C)nc1Cl)=O)NC(c1c(CC)non1)=O c1(CNc2ccc(-c3c(OCC=C)c(OC)ncn3)s2)ccc(F)c2c1CCC2 Cc1cccc(OC(C)C(=O)NCC2CCN(C(c3snc(O)c3Cl)=O)C2)c1 N1(CCN2C(=O)NCC2)CCCC2(CCN(C(C3(C(F)F)CC3)=O)C2)C1 C1(N(C(=O)C(C2CCC(=O)CC2)F)C)CN(C(c2cnc(O)s2)=O)CC12CC2 CCC(C)C(=O)C(=O)N1CC(CCNC(c2ccc(CF)cc2)=O)OC(C)C1 c1(SC)cc(C(N2CCCC(C(C)NC(C3(O)CCOCC3)=O)C2)=O)ccc1F CN1c2ccccc2CC1C(N1CCC(NC(C2CSC2)=O)CC(C)(C)C1)=O CC(C)C1=NOC(CS(=O)(=O)N(C2CCC(NCC3C=CCCN3C)CC2)C)C1 c1(C(N(CC(O)CN(C)C(C2CCCS(=O)(=O)C2)=O)C)=O)[nH]cc2c1CCCC2 Cc1cc2n(n1)CCN(C(C1CN(C(=O)CN3CCCC3)CC1C(C)C)=O)C2 C(CCCCC(=O)NC1(C)CCN(C(=O)C(C)(C)C(C)C)C1)=CCCC C1(C(N2CCN(C(c3c(CC)scc3)=O)CC2CO)=O)CCC(S(C)(=O)=O)CC1 S(=O)(=O)(c1cc([N+](=O)[O-])ccc1Cl)N1CC(C(=O)O)C1c1ccccc1 c1(C(=O)NC(C)CCCNC(=O)CC2CCCN(C)C2)csc2cncn12 C(=O)(CC(C)(C)C=C)NCCCN(C(C(C)OCCC#C)=O)Cc1ccccc1 N1(C(CCC#C)=O)CCSCC1CC(=O)NN1C(=O)CSC1=S Cc1ccc2c(c1)CC(C(N1CCN(C(c3cn4c(n3)CCC4)=O)C(C)C1)=O)S2 N1(C(c2cc(OC)nc(C)c2)=O)CC(C)CN(C(C2(CSC)CC2)=O)CC1C C1(C(=O)NCC(C)(C2CCC2)NC(c2ncccn2)=O)CCCOC1 c1(C(=O)NCC(C2CC2)NC(c2c(C)cc[nH]c2=N)=O)cnnc2ccccc12 c1(CC)cnc(C)c(NC(=O)C(C)(CSC)NC(=O)C(C)NC(=O)NC)c1 CCC(C)C(O)C(C)C(=O)NC(C(N1CCC(OCCOC)CC1)=O)C1(C)CC1 c1(C(N(C(C)CNC(=O)COC)CC)=O)ccsc1 O=C(CCCC1CCC1)NCC1CC(O)(CNC(C2CCOC2C2CC2)=O)C1 C(=O)(C(O)CCNC(c1c[nH]cc1C1CC1)=O)NC1CCN(CCOC)C1 C(=O)(CCC(CF)CF)N1C(C(=O)NC2C(O)C3CCOC23)CSCC1 CC1CCC(CC(=O)NC2CC(NC(=O)C(O)CC3CC3)C2)O1 c1(C(=O)NCC2(OC)CCN(C(=O)CC3CC34CC4)CC2)cc2n(n1)CCCO2 C1(C(N(CC(CCC=C)O)C)=O)CC12CCN(C(c1ccc([N+](=O)[O-])o1)=O)CC2 N1(C(c2cccc(C#C)c2)=O)CC(C)C(N=c2ccn3c(Br)cnc3[nH]2)C1 c1(C(=O)NCC(C)N(C(c2c(C)oc(C(C)C)n2)=O)C)ccc(Cl)c(N)c1 N#CC1C2CC2CN1C(c1cccc(-c2ccco2)c1)=O c1(NC)nccc(C(N2CCCC(NC(C(C)NC(CC)=O)=O)C2)=O)c1[N+](=O)[O-] C1(C(=O)NC2C(C)CCC2C)CCC2(CC2)N1C(=O)CN1CCCC1 c1(CNC(C(C)(C)CCl)c2nnnn2C2CCCC2)ccc(Cl)c(S(N)(=O)=O)c1 C1(NC(CNC(=O)OC)=O)CCC(CNC(c2n[nH]c(C(C)(C)C)n2)=O)C1 C(=O)(C(CNC(=O)Nc1ccccc1)C(C)(C)C)N(C1Cc2cccnc2C1)C CC12CCCC(C(=O)NCCC3(O)CCN(C(=O)Cn4cncn4)CC3)(CO1)C2 C=CC1(CC(=O)N(C(C)C=C)C)CN(C(=O)CC2CC(SC)C2)C1 n1(CC(CC)CC)nc(-c2ccccn2)nc1C1CC1(c1ccccc1)C(C)C CCC(CCC(=O)Nc1cncnc1C)NC(C1CCC(=O)O1)=O C1(C(N2CCC(C(=O)NC3(C(F)(F)F)CC3)(OC)C2)=O)(CC)CC(C)(C)C1 C(CC(=O)NCCc1cccs1)(C(F)(F)F)NC(C(CCC)NC(N)=O)=O CCC(O)CC(=O)NC1C=CCC(C(=O)NCC2CCCC2)C1 C1(NC(c2c(C)onc2)=O)CN(C(c2ccc(C(F)F)c(F)c2)=O)CCC1CO N1(C(CC(C=C)(C)C)=O)CC(C)C(NC(c2ccnc(C(F)(F)F)c2)=O)C(C)C1 c1(C(N2CC(C)C(C(=O)NC3COCCC3(F)F)C2)=O)cccc2occc12 CN1CCC(C(=O)NCC2CN(C(c3c(F)cccc3Cl)=O)CCN2C)CC1=O C1(NC(c2csc(C3CC3)c2)=O)CC(CNC(C2CC2(F)F)=O)C1 CCC(C)(CC(c1nnnn1C)NCCOC(=O)OC)NCc1ccc(C)cc1 c1(C(=O)NC2(C)CCN(C(CCn3c(C)ncc3)=O)C2)cc(N)c(Cl)cn1 Cc1cc(C(=O)NC2CC(CNC(c3occc3F)=O)C2(C)C)ccc1Br C=CCC(CNC(c1cscc1OC)=O)C(=O)N1CCC(C)OCC1 N1(C(c2cc(C)c(C)[nH]2)=O)CC(CNC(C2CC3(C2)CC3F)=O)C2(CC2)C1 C(=O)(CCC(F)(F)F)NCC(CC(N1CCC(CC(C)C)CC1)=O)C C1(CNC(C(CC)F)=O)CCN(C(=O)C(=Cc2cnn(C)c2)C)CC1(F)F N1(C(C(C(C)C)C)=O)CC2CC(C1)C(CO)C2NC(c1nc2ncccn2n1)=O c1(C(C(=O)NC2CCCC2)N(C)CCN2CCOCC2)cc(Cl)cc([N+](=O)[O-])c1 CC(C)C(C(=O)N1CCN(C(c2cnc3ncccn23)=O)C(CF)C1)C(C)C c1(C(=O)NCCCN(C(=O)C(C)(F)CC)CC)cccc(-c2ccccc2)c1 C1(NC(C(=O)N(C(C)C)CC2CCCO2)=O)CC2CCC1C2 Cc1csnc1C(=O)N(CCCNC(=O)CC1(N(C)C)CC1)C1CC1 C1(NC(C=C)=O)CCN(CCC2CC2)C1(C)C C(CCF)(C(=O)N1CC(n2cnnn2)C1)NC(CC(C)C1CC1)=O C(CC)(CC)(CC)NC(C1(S(=O)(=O)N(C)C)CC1)c1n(CCCCCC)nnn1 C(CC(F)F)(C(=O)N1CCC1C(N)=O)N(C)C(C1CCCCC1O)=O N1(C(c2c(-c3c(OC)cccc3)csc2)=O)CC2(NC(=O)C(=O)N(C)C)CCC1C2 Cc1n[nH]c(C)c1CCC(N1CC(NC(=O)C(F)(F)c2cnccn2)CC1C)=O c1(C2N(C)CCC2)ccc(CNc2ccc(-c3ccco3)cc2)cc1 C1(C(=O)NCC2(C(N)=O)CN(C(C3CCCCC3(F)F)=O)C2)CC2(C1)CC(O)C2 N1(C(COCc2n(C)cnn2)=O)CC2CC2(NC(=O)C(c2ccccc2Cl)O)C1 N1(C(Cc2c(C)occ2)=O)CCCC(NC(C2(CO)COC2)=O)C1C N1(C(C2C(CC)CN(C(=O)C(=O)N(C)C)C2)=O)C(CO)CC2CCCC12 N1(c2n(CCCOC)c(C(O)C(C)(C)C)nn2)CCCC2NC(=O)CC12 C(C(=O)NN=c1ccn(-c2ccc(C#N)cc2Cl)[nH]1)OCc1cn(C)nc1 C1(C)(C(=O)NC(C2CCCCC2)C#C)CC2CCC1CC2=O c1(C(=O)NCC#CCNC(C2C(=C)C2)=O)cccc(N)c1 C1(NC(C(CCC)C)=O)CCC2(CCN(C(=O)C3=CCCCC3C)C2)C1 C(C(C)C(C)C(=O)N(C1(NC(=O)CSCc2c(C)noc2C)CC1)C)OC C1(C(=O)NCc2cc(C)c(C(F)F)cc2)CC=CC(N=[N+]=[N-])C1 CCCC(C)C(C(=O)NC1COC1)N(c1c(C)cc(C)cc1C)C C(CCCCC(=O)NCC(C)CN(C)C(C1CC(CCO)C1)=O)SC C1(CN(C(c2cc(CO)n(C)n2)=O)CC)CCCN(C(=O)C(O)C2CC2)C1 c1(C(C)NC(C(C)NC(C2(Cl)C(C(C)=O)C2)=O)=O)cnccn1 C1(NC(C2CCC(C)(F)CC2)=O)CC12CCN(C(c1cc(C(F)F)cs1)=O)CC2 N#CC1CCN(CCCOCCOCCOC(=O)CCC(=O)c2ccco2)CC1 CCCCC(CN(C(=O)CC1CC(F)CN1C(c1cc(C)cs1)=O)C)CC c1(C(C(=O)NCC(C)N(C(=O)C(C)c2cccs2)C)C)ccc(N)cc1 C(=O)(C1Cc2ccccc21)NC1CC(NC(Cc2cn(CC)nn2)=O)C(O)C1 N1(C(CC23C(CN(C(c4c(C)nco4)=O)C2)CC3)=O)CCN(C)C2(CC2)C1 C1(N(C(=O)CC2(C)CCCO2)C)CCC(CNC(=O)COC2CCCC2)CC1 c1(CCC)cc(C(=O)N(CCN(C(c2cn(C3CC3)cn2)=O)CC)CC)n[nH]1 c1(C(=O)NCC(CC)NC(=O)CN2CC3CC3C2)ccc(F)c(Cl)c1N C1(CNC(CCN(C(CCCCNC(C)=O)=O)C2CC2)=O)CC2CCC(C1)C2 C(=O)(C(O)CC(N)=O)N1CCC(C(=O)NC(CC=C)C(=O)OCC)C1 C12(C(=O)NC3C(CNC(CSCCC)=O)CC3)CC(CC)(CO1)C2 c1(CNC(C2(C)CSC2)=O)n[nH]cc1C(N1CCC(OCCO)C1)=O C1(CNC(c2c(C(C)C)onc2)=O)C(C)CCN1C(C1CC(OC(F)(F)F)C1)=O c1(CCCC(=O)NC2CC(N(C(COCCC)=O)CC)C2)ccccc1Cl Cc1cc(=NC2CCN(C(=O)C=Cc3ccccc3)C2)c([N+](=O)[O-])c(C)[nH]1 N1(C(c2cccc(F)c2I)C(=O)NCCSC)CCC(C2=NOCC2)CC1 c1(OC)ccccc1N(C(=O)C#CCNC(=O)CC1CCC(C#N)C1)C N1(C(CCC=C=C)=O)CCC(C2CC2)C1Cn1cc(-c2cnccn2)nn1 C(=O)(C(F)(CNC(=O)C(CC)NC(N)=O)C(C)C)N(C)Cc1ccn(CC)n1 CCC(C)C(C(=O)N1CC2CC1(C(=O)NC1(CC3CC3)CC1)C2)OC c1(OC)cc(C(=O)NCC(CNC(C2(C3CC3)CCC2)=O)CO)ccc1[N+](=O)[O-] c1(CN(CC[Si](C)(C)C)Cc2cn(CCC)nc2)cc(C(=O)O)c(C)n1C C1(OC)CN(C(c2ccoc2CNC(=O)CC2(N(C)C)CC2)=O)CC1O N1(C(C2(C)CC(F)C2)=O)CCOCC(CNC(=O)CC2CC(F)C2)C1 C1(C)(C(=O)NCCN(C(CC2CC(OC)C2)=O)CC2CC2)CCCNC1=O CCCCC(O)CC(=O)NCC(C)(CC(C)C)NC(c1cc(C(N)=O)cn1C)=O c1(CN2CCC(NC(c3ccc(SC)cc3)=O)C2C)cnc2c(c1)NC(=O)CO2 c1(OC)cccc2c(N3C(C(=O)N(C)Cc4cccnc4)CC4CC34)ncnc12 c1(C(N2CCC2CC(=O)NC(CN2CCCC2)CO)=O)c[nH]c2ncccc12 O(N(C)C(=O)C(CNC(=O)C(C)C(C)C)C(C)(C)C)CC(=O)OC C(=O)(C1CSc2ccccc21)N(CCCN(C(c1ccc(C#C)cc1F)=O)C)C CC(C)(CC(F)C(=O)NCC(O)C(N)=O)NC(c1coc(CO)c1)=O Cc1noc(CCCC(=O)N2CCC(CCNC(C3CCC3)=O)C2)n1 c1(C(=O)NCCN(C(c2c(SC)csc2)=O)C(C)C)sc(-c2nc[nH]n2)nc1C C=CCC(CC(=O)NC(CC1CC1)CC1CC1)NC(c1ccc(C)nn1)=O c1(C(=O)NC2(CNC(C3CN(C)C(=O)C3)=O)CCC2)cnn2cc[nH]c12 C(=O)(C1=CCCCCC1)NCC(C(=O)N(C)Cc1nc(C)sc1)CC1CC1 C1(NC(C(C2(OC)CCCC2)(F)F)=O)CN(C(=O)COC(F)F)C2(CCOC2)C1 c1(C(N(CC(CNC(c2[nH]cc(C)c2)=O)(C)C)C)=O)cc(F)c(F)cc1O C1(C(=O)OCC(=O)Nc2c(OC)cc(OC)c(Cl)c2)CC(C2CCCCC2)C1 c1(C(=O)NCC(CN(C(C(CC)N2CCCC2=O)=O)C)O)ccc(Cl)cc1CC C(=O)(CCCC(F)(F)F)N1CC(OCCNC(CC(CC)SC)=O)C1 CCC(CC(=O)N1CC2CC1C2NC(=O)C(C)Cc1cnc[nH]1)CC(C)C c1(C(N2CCC(Oc3ccc(OC)cc3)C2)=O)ccc2c(c1)NC(C)CC(=O)N2 C1(=CC(=O)N(CCN(C(=O)CC2(C)CC2(F)Cl)C(C)C)C)CCN(C)C1 c1(C(=O)NCC(C)N(C(=O)CNC(=O)CC(F)(F)F)C)cc([N+](=O)[O-])ccc1Cl CC1CC(N)CCN1Cc1ccc(F)cc1Br N1(C(C2(NC(=O)C=CCN3CCC3)C(C)C2)=O)CCOCC(C)(F)C1 C(=O)(CC(O)C(C)C)NCCC(CNC(c1c(C)coc1C)=O)O c1(N(C(C)C(CCN=O)=O)C(c2ncnc(C)c2C)=O)c[nH]c2nccc-2c1 N1(C(CC2(COC)CC2)=O)CCC(C(=O)NC2CC(O)C(O)C2)C1C(C)C N1(C(C2C(c3c(C)ccs3)C2)=O)CC(CN(C)C(c2cnnn2C)=O)C2(CC2)C1 CCC(CC(=O)NC1CN(C(=O)C(OC)OC)C(C)(C)C1)C(F)F N1(C(c2c(CC)cco2)=O)CCCCC12CN(C(=O)CN1CSCCSC1)C2 C(=O)(NNC(=O)C(C(=O)OC(C)(C)C)(C(F)(F)F)OC(C)(C)C)C1C(=C)C1 Cc1nc(C)c(CC(=O)NCCCN(C(=O)C(O)C2CCCC2)C(C)C)s1 C=CCCCCC(=O)N1CCCC(CO)(NC(=O)C(C2CCCC2)OC)C1 C1(C(=O)NCCOCC(N)=O)CCN(C(=O)C(F)CC2CC2)C12CCC2 C1(NC(=O)NC(c2ccc(C)o2)C2CC2)CCCCC1c1nc[nH]n1 C1(OC(C2C(CC=C)CCC2)=O)CCOC2(CCOCC2)C1 N1(C(=O)Nc2c(Oc3cccc(C)c3)nccc2)CC(F)(F)C2(CCCC2)C1 C1(NC(c2nc3nccc(C)n3n2)=O)CCCC2CN(c3ncc(Br)cn3)CC12 c1(SC)cccc(C(=O)NCC2COCCN2C(=O)C(C(C)C)C2CCC2)n1 CN1CC(O)CC1(C)C(=O)NCC=C1CCN(C(=O)CCn2ccnc2)CC1 N1(C(=O)CC2CCN(C(c3c(O)cccc3O)=O)C2)CCC2(CCCO2)C1 C1(CNC(C2C(OCC)C2)=O)CC2(CC2)CN1C(c1ccnn1C(C)C)=O c1(C(=O)NC2CC(C)CN(C(=O)C(=O)NC3CC3)C2)ncn2cc(Cl)ccc12 C(=O)(C(F)(F)C(C)(C)O)NCC(CC)NC(c1ccccc1-n1cccc1)=O c1(C(N(C2CCC(NC(=O)C(O)CC(C)(C)C)C2)C)=O)ccc(F)c2occc12 N1(C(c2ccc(C(C)C)cc2)=O)CCC2C(NC(=O)CSc3nc[nH]n3)C2CC1 CC(C)C(O)C(C)C(=O)NC1(C(=O)NC2C3CCC2CC3)CC(O)C1 C1(CC)(NC(=O)CC2(CO)CCOCC2)CCCN(C(c2csc(Cl)n2)=O)C1 c1(OC)cc(NC(C)=O)cc(C(N2CCC(N(C)C(C34CC(O)C3C4)=O)C2)=O)c1 CC1CN(C(C2CCN2C(C)(C)C)=O)CC1C(=O)NOC1CCCCCC1 C1(NC(CNC(C)=O)=O)CCC12CCN(C(=O)C(c1ccn(C)n1)C)CC2 N1(C(CCNC(CC(C)C)=O)=O)CC(NC(C2(C(F)F)CC2)=O)CC(C)(C)C1 CC(N=[N+]=[N-])C(=O)NCCSCC(=O)NCC1CC1(Cl)Cl n1(CC(N2CCCC(OCCC)C2)=O)c2ccccc2c2ccccc12 N1(C(CC(C)C(F)F)=O)CCCC2(CCN(Cc3nnc(C4CC4)s3)C2)C1 C(=O)(CCCCC#N)NC(C(C)NC(c1noc(C)c1Br)=O)C(C)C N1(C(C=CC=CC)=O)CC2CC(NC(=O)Cc3ccc(F)cc3CC)CC1C2 C1(N(C(C2CCC(CC)C2)=O)C)CCN(C(=O)CCNC(=O)COC)CC1 C(CCCCCCC(=O)N1C2CCC1CN(C(=O)CC(=O)NC1CC1)C2)SC C(=O)(C(O)CC(C)(C)C)NC1C(NC(CC(CCSC)O)=O)CCC1 CCCCC(CN=c1[nH]cnc2ccccc12)NC(=O)C(F)(F)C1CC1 C(=O)(CC1=CCN(Cc2ccccc2)CC1)Nc1c2ncn(C)c2ncn1 C1(C(=O)NCC2COCCN(C(C(CC)F)=O)C2)C(C)(C)CCCC1(C)C N1(C(c2c(C(C)NC(=O)CN=[N+]=[N-])noc2)=O)CCSCC(C)C1 Cc1cc(C(=O)NCC2CCCC2(C)CN(C(=O)CC2CN(C)C2)C)sc1Cl C=C1CC2(C1)CC(C(=O)NCC1(C(N)=O)CN(C(c3ccnc(C)n3)=O)C1)C2 C1(C)(C(=O)NC2C(C(N(CCCCO)CCCC)=O)C2)CC1(F)F c1(NCC23CCC(NC(c4cc(C)c(C)[nH]4)=O)(C2)CO3)ncc([N+](=O)[O-])cc1Br c1(OC)cccc(Cl)c1CNC(N1CCNC(Cc2ccccc2)C1)=O C1(NC(=O)C=C2CCCCC2)CCN(C(=O)CCc2nc[nH]n2)CC1O c1(CC(=O)OCC(c2cccc(Br)c2)C)ccc(C(F)(F)F)nc1 Cc1cc(-c2cn(C3CC4(C(=O)NCCCCCCCO)CC34)nn2)cc(F)c1 N1(C(Cc2cccc(N)c2)=O)CCC2(CCCCC2NC(c2c[nH]nc2F)=O)C1 C1(C(N(C2CCN(C(c3ncnn3CC)=O)C2)CC#C)=O)CC(C)(C)CN1C c1(C(N2CCC(C)(NC(c3n(C)ccn3)=O)C2)=O)ccc2c(c1)CCNC2=O N1(C(c2cc(C)no2)=O)CCC(CC(=O)NCC2CCN(C(C)C)C2)C1(C)C C1(CC(=O)NCC(C)(C2CCC2)NC(c2n(C=C)ncc2)=O)CCCCC1(C)C c1(C(=O)NC2CCC(NC(=O)CCF)C2)ccc(C(F)(F)C(F)F)cc1 c1(CC(=O)NC2(C)CN(C(C(C)NS(C)(=O)=O)=O)C2)cccc2ccoc12 C1(NC(C(COC)C)=O)(CNC(=O)CCn2c(C)ccc2C)CCOCC1 c1(CN2CCN(C(Cn3ncn(C)c3=O)=O)CC2)cnc(N)c(Cl)c1 C(=O)(C(C)CCC(C)(C)C)N(CCC(=O)NCCNC(C(C)C)=O)CC1CC1 c1(C(=O)NCCNC(C2CCCS2)=O)ccc(OC(F)F)nc1 C1(N(C(c2cn(CC3CCCO3)nn2)=O)CC)CCCN(C(=O)C(N)=O)CC1 c1(C(=O)NC2CCN(C(c3ccc(C4CC4)o3)=O)C2)cncc(OC(F)(F)F)c1 C1(C(=O)N(C)CCc2ccccn2)(CC)CCN(C(c2ncncc2N)=O)C1 N(C1CCCc2c[nH]nc21)C(CC(CNC(c1c(C)n[nH]c1)=O)O)=O c1(C(=O)NC2(CCCNC(CC(C)c3ccco3)=O)CC2)noc2c1CCCC2 Cc1nc(C2CC2)ncc1C(N1CCN(C(c2cnc(O)s2)=O)C(CCO)C1)=O C(C1CCN(C(C2CC3CCC2O3)=O)CC1)=CC(=O)Nc1ccc(C(C)C)nc1 C(C1c2ccccc2CCN1C(c1c(C)nsc1C)=O)NC(C(C(CC)C)C)=O c1(C(N2CC3CCN(C(CC(CC)CC)=O)C3C2)=O)cnc2c(c1)NCC(=O)N2 c1(CNC(C(C)(CO)NC(c2cc(CO)on2)=O)=O)ccc(F)nc1F c1(C(N2CC=C(CNC(Cc3n(C)ccn3)=O)CC2)=O)cc(P(C)(C)=O)cs1 CCCC(CC)CC(=O)N(C1CCN(C(=O)CC2(O)CCOCC2)C1)C c1(C(C)C)nc(NCc2cccnc2OCC(F)F)cc(=NCCS(C)=O)[nH]1 C1(C(N2CC3=C(CN(C(CN(CC)CC)=O)C3)C2)=O)CCC2C(CC1)C2(F)F C1(C2CCN(C(c3ccsc3C(F)F)=O)CC2)(NC(c2ccsn2)=O)CC1 N1(C(CN(C2CC2)CC)=O)CCC(NC(=O)C(c2cccs2)SC)C1C1CC1 CCCC(O)CC(=O)NC(C1(O)CN(C(=O)Cc2cccc(Cl)c2Cl)C1)C N1(C(C(n2ncc(C)c2)C)=O)CCc2sc(-c3ccnc4[nH]ccc34)nc2C1 Cc1cc2c(cc1C)C(C(=O)N(C1CCN(CC=CCl)CC1)C)CO2 C(CCC(O)C(=O)NC(C)(C)CC1CCOC1)NC(Cc1c(C)ncs1)=O N1(C(=O)NC(c2csc(Br)c2)C)CCS(=O)CC1c1cnn(C)c1 c1(CC)ccc(N)c(C(N2CC(NC(=O)C(C)CCOC)C(O)C2)=O)c1 c1(C(=O)NC23CC(COCCOC)(C2)C3)[nH]nc2ncccc12 C(CCC(C)C)(C(=O)NC1C(CNC(=O)Cc2sc(O)nc2O)CCCC1)OC O=C1CCc2cc(C(N3CCC(CNC(=O)C4CC4)CC3)=O)ccc2N1 N1(C(C2=CCCC2C)=O)C2CCC1CN(C(=O)CCc1cn[nH]c1)CC2 CC1CCN(C(=O)CN2CCC(C(F)(F)F)CC2)CCN1C(C12CC(F)(C1)C2)=O N1(C(C2CCS(=O)(=O)C2)=O)CCN(C(=O)CCn2ccccc2=O)C2COCC12 C1(C(N2C3C(NC(CC(N4CCCCC4=O)C)=O)C(C3)C2)=O)CCCCNC1=O n1(CC(=O)N(CC(CO)(CO)NC(C(C)=C2CC2)=O)C)nc(C)c([N+](=O)[O-])c1C CC1CN(C(c2ccsn2)=O)CC(C)C1NC(c1c[nH]cc(Br)c1=N)=O C1(C(=O)NCC2(O)CN(C(CC3ON=C(C)C3)=O)C2)CC(C2CC2)C1 Cc1ccc(C)c(C(N2CCC(=CCNC(C3CC(C)C3)=O)CC2)=O)n1 C1(C(=O)NC2CCCC(C#C)C2)CC2(CCN(C(c3cn(CC)nc3C)=O)C2)C1 C1(CC(=O)NC(C(=O)NC2C(CC)C2)C2(C)CC2)CCCN(C)C1 O=C(CCC(=O)N1CCC1CNC(C12CC(C1)C(c1ccccc1)O2)=O)C1CC1 c1(NS(N(C)C(COC)C)(=O)=O)nc(Cl)ccc1O c1(C(=O)NC2CN(C(C(OC)OC)=O)CC2SC)cnc2ccc(F)cn12 C=CCC(CNC(=O)C1=CC(C)(CC)C1)C(=O)NC1CC(CO)N(C)C1 C1(OC)CC(C)CN(C(C2CC(F)(F)CN2C(=O)CN2CC(C)(C)C2)=O)C1 c1(C(=O)NC2C(C)CN(S(C)(=O)=O)CC2)ccc2c(c1)CNC2=O C(=O)(N=c1ccnc(Br)[nH]1)C1N(Cc2c(O)ccc(C)c2)CCOC1 C1(C(N2C(c3cn(C)nc3)CSCCC2)=O)CCC(C)(C(=O)O)C1(C)C N1(C(C2(C=C)CC2)=O)C2CCCC1CN(C(c1cnc(C(F)F)cn1)=O)C2 c1(C(N2CCC(Cn3cc(C(C)(C)OC)nn3)C2)=O)ccc(F)nc1 N1(C(C(CC)n2cncn2)=O)CC(NC(=O)CCc2cnco2)CC(C)(C)C1 C1(C)(CNC(Cc2cc(C)ns2)=O)CCCN1C(=O)CC(C1CC1)C1CC1 C1(N)CCC12CCN(C(=O)C(F)(F)F)CC2.CC1(C)CN(CC(O)CO)CCC1O C(CNC(c1ccnc(OC)n1)=O)(CC(=O)N1CCC1C(N)=O)OC C1(C(N2CCC(C#C)(F)C2)=O)CN(C(=O)CCc2cnc(C)o2)C2(CCC2)C1 C1(CNC(c2c(C)nco2)=O)C(C)CCCN1C(C1CCC2CC2C1)=O C1(CN(C)C)CC2CC2N1C(=O)CCc1cn(C)cn1.C12CCCN1C2=O Cc1ccc(C)c(C(N2CC3CC3(CNC(=O)CN(C3CCC3)C)C2)=O)c1C C=CC(C)CC(=O)NCCCCNC(=O)CCC1CCC1 C#CC1CN(C(=O)C=CCC2(NC(c3cc(OC)cs3)=O)CCC2)CCN1C Cc1nc(C=CC(N2CCC3(NC(=O)CSCC(F)(F)F)CC3C2)=O)[nH]c1C c1(C(=O)NC(C(N2C(CCC)CCC2)=O)Cc2ccco2)cc(F)n(C)n1 N1(C(c2cnn(C)c2)C(=O)NCCC)CCc2c(C(=O)NC)csc2C1 C1(n2cc(C(C)(C)OC(=N)O)nn2)CC2CCC1(NC(c1ncccc1Br)=O)C2 N1(C(C=Cc2cn(C)nc2)=O)CCC2(CC1)CN(C(=O)CCN1CCC(F)C1)C2 C1(C(N2CCN(C(c3ccncn3)=O)CC2)=O)CCCCC12CC2(F)F c1(C(N(CC(C)NC(CCCCCC)=O)C)=O)ccc(N)c2ncccc12 CCCC(CNC(C1(Cl)CC1C(C)=O)=O)C(=O)N1CCCC1CN=[N+]=[N-] Cc1c(C(N2CCCC(NC(=O)C(O)CCC(C)C)CC2)=O)[nH]c2ccccc12 c1(C(N2CC(CNC(CC3CCC(C)C3)=O)C2)=O)cc2nc(Cl)ccc2o1 C1(N(C)C(c2ccc(C(F)F)o2)=O)CCN(C(C2CC2(C)C)=O)CC1 C1(NC(C2CC(N(C(=O)CC3C=CCCC3)C)C2)=O)CCCC(C2CC2)C1 CNS(=O)(=O)NCC(N1CCCC1C(C)(C)CNC(C1(C)CCOC1)=O)=O C1(C(N2CCCC(OC)C2)C(=O)NCC(C)C)C2(CCC2)C12CCC2 c1(C(N2CC3C(NC(C4(C#N)CC4)=O)(CCC3)C2)=O)cccc2cc(Cl)ccc12 c1(COC(=O)NCCCOC2CCOC2)ccc2c(Cl)nccc2c1 C1(CC(=O)NCCCSCCO)CCCN(C(c2cncc(C3CC3)c2)=O)CC1 c1(C(N2CC3C(CNC(c4nc(C)oc4)=O)C3C2)=O)cccc2c1CCN2 CC1(C)COC(CC(N2CCCC2CCNC(c2ccn(C3CC3)n2)=O)=O)CO1 Cc1ccc(C(N2CC(CC(C)NC(=O)Cn3cc[n+](C)c3)C2)=O)c([N+](=O)[O-])c1 c1(C(=O)NC2C3CC2N(C(c2cnco2)=O)C3)ccnc(O)c1Br Cc1ncsc1CN(C(C1CC2CC2C1)C(=O)NC1CCCC1)C c1(C(=O)NC2CCCN(C(c3nc(Br)c[nH]3)=O)C2)noc2ccc(Cl)cc12 c1(C(=O)NC2(CNC(CC(C)(C)F)=O)CCC2)oc2ccccc2c1CN(C)C c1(CN2C(C(=O)Nc3n(CC)nnn3)CC3CC32)cc(Cl)cc(Cl)c1Cl C1(CNC(CC2(C)CC2(Cl)Cl)=O)CC2(CC2)CN1C(=O)Cc1n[nH]c(=N)s1 C1(CC)CCOCCN1C(=O)C(C1CCCN(C(=O)CCC(C)(C)OC)C1)(C)C Cn1cc(N(C(=O)Cn2nnc(=N)[nH]2)C(c2ccccc2)(C)C)c(OCC(F)F)n1 Cc1ncc(N)cc1C(N1CCC(NC(=O)CCc2cnn(C)c2)C(C)C1)=O N#Cc1csc(C(=O)NCC(c2ccccc2)CNC(c2occc2Cl)=O)c1 C12(C(=O)NC(CC(C)NC(C3CCN(CC4CC4)CC3)=O)C)CCOC(C)(C1)C2 Cc1cn(C)nc1CNC(C1CC1Cl)=O.c12cn(nn1)CCONC2=O Cc1nccc(C(=O)NC(CNC(C2(C(C)C)CCC2)=O)C(C)C)n1 CCCCCCC(F)C(=O)NCCCN(CCCCNC(=O)C(CC)OC)CC C1(CC(=O)NC2C(NC(=O)CCc3cc[nH]n3)CCC2)CC2(CCCC2)CO1 N1(C(C2C(C)(C(F)F)C2)=O)CC(NC(=O)CSC2CC2)C(CC2CC2)C1 N1(C(C=CC(C)(C)SC)=O)CCCN(C(=O)Cc2cn(C)nn2)CC1 c1(C(N(CC(C)NC(C2(CC(F)F)CC2)=O)C)=O)cscc1Br N1(C(C=CCC)=O)CCCCC2(CCN(C(=O)C(c3ccc(C)o3)C)C2)C1 c1(C(=O)OCCNC(C(COC)N(C)C)=O)c(O)cccc1O.C(CC1CC1)O N1(C(CC2CCCN(C(C(COC)OC)=O)CC2)=O)CC2CC(C1)C2(C)C N1(C(c2c(C)cncc2C)=O)CCC(C2(NC(=O)C(C)N(C)C)CC2)CC1 O=S(=O)(c1ccc(NCCOCCC2CC2)c(Br)c1)NC1CC12CCCC2 C1(N(C(=O)CCc2nccs2)C)CN(C(C2CC(F)C2)=O)CC1F Cc1cnc2c(C(=O)NC3CC(CNC(=O)CN(C)C(N)=O)C3)c(C)nn2c1 C1(N(C(CC)=O)CC2CC2)CCN(CCCn2cc(C(C)O)nn2)C1 N1(C(CC(C)SC)=O)CC(NC(=O)CCN2CCC(F)C2)C(CC2CC2)C1 c1(C(C)NC(CCCC)=O)ccc2c(c1)CN(C(C1CCOC1CC)=O)C2 c1(C(N(CCOCC)C)=O)c[nH]nc1CNC(=O)Cc1ccco1 N1(Cc2nc(C)n(C)n2)CCC(O)C(C(=O)NC2(C3CC3)CC2)C1 c1(C(=O)NC23C(CN(C(CNC(N)=O)=O)C2)C3)scc2c1OCCO2 c1(CC(=O)NC(CC)(C)CNC(=O)COC(F)(F)F)ccc(C)c(OC)c1 c1(CC(=O)NC2(NC(c3ccc(C(N)=O)o3)=O)C(C)C2)cccnc1.C1(C)CC1 C1(C(=O)NC(CC#C)CC#C)CC2CCC(C1)N2C(=O)C(C)(CC)CC C12(CNC(=O)CN3CC=CC3)CCCC1N(C(=O)CN1CC=CC1)CCC2 N1(C(C(C)CC2CCCC2)=O)CCC(C(=O)N(C)CCN(C)C)C12CCC2 Cc1cnc(C(=O)NC2C=CCC(C(=O)Nc3cncc(Cl)c3)C2)c[n+]1[O-] c1(OCCOC)ccc(C(=O)NC(C)CCNC(=O)C(F)=CCCF)cc1N CCC(C)(O)C(=O)NC1CCC(CNC(C2(c3cncnc3)CCCC2)=O)C1 Cc1cccc(CC(=O)NCC(C(C)(C)C)NC(=O)CSC(=N)N)c1 Cc1cnc2n1CC(C(=O)NCC(O)CNC(C1(S(N)(=O)=O)CC1)=O)CC2 CCCCC(C(=O)NCC(C(=O)NCCCc1ccco1)C(C)C)N(C)C c1(C(=O)NCC2CCC(CNC(C3(C)ON=C(C)C3)=O)CC2)cccc(Cl)c1C C1(CC(N2C(C(C)NC(C3(CF)CCC3)=O)CCC2)=O)CC(C)(C)OC1=O c1(C(=O)NC(c2nncs2)C)ccc2c(n1)CN(C(C1(C)COC1)=O)CC2 c1(OC)ccc2c(c1)C1(CCO2)CC1C(N1CC(CC(=O)O)C(O)C1)=O C1(O)(CC(=O)NC2(C)CC(NC(=O)C(c3cccc(F)c3)O)C2)CCOCC1 C12(C(=O)NCC3C(C)CN(C(=O)C(C)(C)CO)C3)CC1COC21CCC1 c1(NC(C(CNC(CCN(CCOC)C)=O)C)=O)ccc(F)c2c1CCC2 C(C(CC(F)(F)F)NC(=O)Cc1cnc[nH]1)NC(c1c(C)sc(C(F)(F)F)n1)=O n1(CC)cc(CN(C)C(C2(CNC(c3cc[nH]c3)=O)CCCO2)=O)cn1 C1(NC(c2ccc(OCC#C)cc2)=O)CC2CC1CN(C(=O)COC(C)=O)C2 N1(C(C(C)C2CCC2)=O)CCC(O)(CN(C(=O)C=Cc2ccoc2)C)C1 c1(OCC)c(F)c(C(=O)NCC(C)NC(=O)C(C)=C(C)C)cc(F)c1F c1(CC(CC)NC(=O)C(=O)N(C2CCC2C)C)ccccc1 c1(CC(=O)N(c2ccc(Br)nc2)C)csc2c(F)cccc12 Cc1ccccc1CC(N1CCC(C(C)NC(=O)CCc2ccccc2C)C1)=O C12(NC(c3n(C)cc(Cl)c3)=O)CCCC1CN(C(C1CCCC1(F)F)=O)C2 CC1(C)CCCC(C(N2CCCC2CNC(c2cnc(C(F)(F)F)cn2)=O)=O)O1 C1(CC(=O)N(CCCNC(c2coc(C3CC3)n2)=O)CCC)CC(=O)NC1=O C1(NC(C(CC)=CCCC)=O)CCOCC1C(=O)NOCC1(C)CC1 c1(-n2cc(CCC(=O)NCC(=O)NCC#C)nn2)cc(Cl)c(Cl)nc1C [N-]=[N+]=NC1CN(C(c2cnc3c[nH]nc3c2)=O)CC1NC(C1(F)CCCCC1)=O N1(C(c2c(CC)cccc2C)=O)CC(C)C(NC(=O)CC(C)=C(C)C)C(C)C1 Cc1cccc2c1OC(C(=O)NCC1CCCN(C3CCSC3)C1)C2 CCCCCC(O)CC(=O)NC1CCN(C(=O)C(O)C(C)CC)CC1C(N)=O N(C(=NCc1ccnn1C(F)(F)F)NCC(C)(C)C(C)(F)F)C(C)C CCCCC(O)C(C)C(=O)OC(C(C)(C)CC)OC.c12ccccc1O2 C(C1CN(C(=O)C=C(C)C)CC1C(=O)NCCN(C)CCF)=CC c1(-n2cc(CNC(CC3(OC)CCCCC3)=O)nn2)ccc2c(c1)OCCO2 C1(N(C)C(c2sccc2Cl)=O)CCN(C(c2cc(C#N)cs2)=O)CC12CC2 C12(C(=O)NCCOCC(=O)O)COCC1C2(F)F.c12cccc(c1)-c1cn(nn1)C2 C(C1COC(C)(C)O1)=CC(N1CCCC(C(=O)NCCc2ccn(C)n2)C1)=O N1(C(C2C(C)(C)CC2)=O)CCC2(CC1)CC(NC(C1(O)CC3CCC1C3)=O)C2 N1(C(C(C)SCC)=O)CCC(NC(C2CCC(F)(F)CC2)=O)C(CO)CC1 N1(C(C2(CNC(=O)CCCn3ccnc3)CC(=C)C2)=O)CCC2(CCN(C)C2)C1 C#Cc1ccc(C(=O)N(C2CCN(C(c3cc(SC)nn3C)=O)CC2C)C)cc1 C1(C(=O)NCc2c[nH]c(CN3C4CCC3CC4)c2)CCCC(OCCOCCO)C1 c1(C(N2CCCN(c3snc(CC)n3)CC2)C2CCOC2)cccc(C)c1C N1(C(CC2CN(C(C)=O)C2)=O)CC(O)(C(C)NC(C2CNC(=O)O2)=O)C1 CC1CSCCN(C(C2CCN(C(=O)C3CC(=O)C3)O2)=O)C1 CC1(C)CC1(C)NC(N)=O.C1(C)(CCN2CCCCC2)c2nnnn2CCN1 N1(CCN(C)C(C2CCCC2)=O)CCN(C(C2OCCC2(C)C)=O)CC1 N1(C(CCc2c(C)nn(C)c2)=O)CC(C)(C)CC1CNC(=O)C=CC1CCCO1 N1(C(C2(C)CC2)=O)CCCN(CCNC(c2ncc(F)cc2F)=O)CC1 c1(OC)cc(C(c2nnnn2C(C)C)NCC2CCCC(C)(C)C2)c(F)cn1 C1(F)(C(=O)NC2C(C(=O)NCC3C(C)(C)OCC3)CCC=C2)CCCCCC1 C12(CNC(C(CC)CC)=O)CCCCC1CN(C(=O)C#CC(C)C)C2 c1(OC)nc(=NCC2CCCC(NC(=O)C(C)CC3CCCC3)C2)[nH]c(C)c1F O=C(C1=CCCCO1)NC1CCCN(C(C23COCC(C2)OC3)=O)CC1 c1(C(=O)OCc2cnccc2C)cc(NC(C)=O)cc(N2CCCC2=O)c1 C(CCCCCC(=O)NCc1cncc(OC)c1)NC(C(CCC)OC)=O N1(CC)N=C(C(=O)NC23CC2CN(C(c2cnn(C)c2C#N)=O)C3)CCC1=O S(=O)(=O)(c1cccc(F)c1)NCc1occ(C(=O)Nc2ccc(C)cc2)n1 C=CCC(C(=O)N1CCN(C(=O)CCOCCC(F)(F)F)CC1C(C)C)C(C)C c1(C(=O)NCC(C2CCCO2)O)ncoc1CNC(c1ccnn1C(F)F)=O c1(C(C)=O)ccc(C(=O)NC(CNC(=O)CC2(C)CC2(F)Cl)C(C)C)s1 C1(NC(c2c(CC)cns2)=O)CN(C(=O)COC(C)(C)C(F)(F)F)CCC1(C)C CC1=CCC(C(=O)NC(C)C(=O)NCC(O)CN(C)C)CC1 c1(COC)ncccc1C(=O)NCC1(NC(=O)C(C(C)O)NC(=O)C2CC2)CC1 CC1CCCC=C1C(=O)NCC1CCCN1C(c1cc(O)ccc1Br)=O c1(CONC(C2CC(F)(F)C2)=O)nc2ncc(Br)cc2o1 C1(C(=O)NCc2ccoc2)N(C(C2CC2C2CCC2)=O)CC12CCCC2 N1(C(c2cn(CCC)nc2)=O)CC2(C1)CN(C(=O)CC(C)(C)CC)CC2C(=O)O C1(C(=O)NCC2CC(NC(C3CCC(F)CC3)=O)C2)CCn2ccnc2C1 CP(C)(=O)C1CCCC1C(N1CCC2CN(C(=O)CSCc3cscn3)CC12)=O C1(C(N(C)CC2(O)CN(C(=O)CC3CC(=O)C3)C2)=O)CC(c2ccccc2)=NO1 C(=O)(C(C(C)(C)C)NC(=O)C(c1ccn(C)c1)C)NC(COCC)CO C(CNC(=O)C(C)(C)c1ncco1)(CC(F)(F)F)NC(c1cc(CC)[nH]n1)=O N1(c2snc(CC)n2)CC(NC(=O)C(C2CCOC2)OC)CC2(CC2)C1 C1(CNC(c2cc(C)on2)=O)CCCCN(C(=O)COCC(F)F)C1 c1(C(=O)NCC(C)(C2CCC2)NC(CC2(C)OCCO2)=O)nccc2nn[nH]c12 CCC#CC(C)(C)NC(=O)C=CC(C)(C)NC(=O)CC(C)(F)F Cn1ccc2ccc(C(=O)NC3(C)CCCN(C(=O)CS(=O)(=O)C4CC4)C3)cc12 N1(C(=O)Cn2ccnn2)CCCC(F)(CNC(C2(CO)CC(F)(F)C2)=O)C1 N1(C(c2ccc(CN=[N+]=[N-])o2)=O)CCC2(C1)C(F)(F)C2(F)F c1(OCC)ncc(F)c(=NCCC(=O)N(C)Cc2ccc(F)cc2)[nH]1 CCCCCC(C)(C)C(=O)OC.C(=O)(CC(C)CC(=O)C12C3CC1CCC32)C=O.OC c1(C2C(C(N(CCCNC(C3C(=C)CC3)=O)CC)=O)CC2)nc(S)n[nH]1 C1(C(=O)NC(C(C)(C)C)CO)CCC2(CC2)N1C(C12CCC(C1)C2)=O CC1CC(NC(C2(CO)COC2)=O)CCN1C(=O)C(Cc1ccccc1)C1CC1 C1(CNC(CCc2cc(C)no2)=O)C2CN(C(=O)C(C)NC(=O)C3CC3)CC12 Cc1cc(C(=O)NCC2CCC(NC(=O)C(F)(F)C(O)C3CC3)C2)cc(Cl)n1 C1(C(=O)NC(CNC(c2cncc(C)c2)=O)CO)CC2(CCCCC2)CO1 CCC1=C(C(=O)N2CCC3C(C(=O)NCCC4CC(C)C4)C3C2)CCCO1 c1(CCNC(C2CCCN2C(=O)CCc2nncs2)=O)ccc(F)nc1 CCCC(C)(O)CC(=O)NCC1CCCN(C(=O)CNC(c2cnccn2)=O)C1 N1(C(c2cc(CCC)[nH]n2)=O)CCCC(O)(CNC(c2[nH]c(C)nc2CC)=O)C1 C1(CNC(c2nnnn2C2CCOCC2)C(C)C2CC2)CC12CCC(O)CC2 C1(C(=O)NC(C)CN(C)C(C2CC3COCC3C2)=O)(OC)CCC(C)(C)CC1 C#CCC(O)C(=O)NCC(C)NC(c1ccc(C(C)=O)cn1)=O c1(OCOC)ccc(C(N2CCC(C)C2CNC(=O)CCc2cnc[nH]2)=O)cc1 N1(C(c2cc(OC)nc(Cl)c2)=O)CC2(CCN(C(=O)CC3(C#N)CCC3)CC2)C1 C(=O)(C1=CNC2=NCCC2=C1)N1CN1.CC1(C)CN(CC(N2CCOCC2)=O)C(C)(C)C1 CCCC(C#N)C(=O)N1CC(CC(=O)NC(C)(C)CC(F)(F)F)C(C)C1 C1(CNC(C2N(CC)CCCC2)=O)CCN(C(=O)C(C)(C)C(=O)N(C)C)CC1O CC1NC(=O)OC12CN(C(C1(NC(C3CC=CCC3)=O)CCCC1)=O)C2 c1(CC)cnc2ccccc2c1C(=O)NCC1CCC(NC(=O)C(Cl)=CCl)CC1 C1(NC(C2(CC)COC2)=O)CN(C(C2CCCOC2)=O)CC(C)(C)C1 C=CCCCC(=O)N1CC(C(N2CCC(C)(CC)C2)=O)(SC)C1 c1(C(CC)(C)C)cn(Cc2cc(C(=O)NC3(C(F)F)CCC3)on2)nn1 C=CC(O)C(=O)NCC(O)CCNC(=O)Cc1csc(C(F)(F)F)n1 C(=O)(C1Cc2ccccc21)NC(CC)CNC(=O)C(F)(F)c1ccsc1Cl C(=O)(C(F)(CNC(C1CC(F)(CF)C1)=O)C(C)C)Nc1c(OC)cc(C)cc1 C1(CNC(C=C(C)Cl)=O)CCCC(N(C)C(C2(C(=O)NC3CC3)CC2)=O)C1 c1(C(C)NC(=O)Cc2ccc(C(=O)OC(C)(C)C)cc2)ccc2c(c1)CCN2 c1(C(NOCC(=O)NCC2(COC)CCCC2)=O)cccn2ccnc12 n1(CC)cnc2[nH]c(=NC3CCS(=O)C3)nc(N3CCCC(S(C)(=O)=O)CC3)c12 C(=O)(CC(C)CC(C)(C)C)NC1CCCN(C(c2cc(OC)ncc2Cl)=O)C1 N1(C(c2ncn(C)c2)=O)CC(NC(=O)CC2(C)CCOC2)C(n2ccnn2)C1 C(=O)(C(C)(CCC)CCC)N1C(C)CCN(C(CCCC)=O)CC1 N1(C(C(C(C)C)=O)=O)CCC(CC(N2CCN(CC(N)=O)CC2)=O)C1(C)C c1(OCC#N)cccc(NC(=O)CC2COC3CC2C3)c1 N1(C(=O)CC2C=CCCC2)CC2CCC(C1)N2C(c1cc(CN(C)C)c[nH]1)=O C1(C(=O)NC(CCCC)CC)CC2(CCN(C(C3CCCC3OC)=O)C2)C1 CC(C)C(C)CC(=O)N(CC(C)(C)C(N1CCOCC(CO)C1)=O)C c1(C(=O)NC(C(=O)N(CCCO)CC)COC(C)C)ccc(C)c(C)c1F c1(C(N2CC3(CC(CNC(C(C)CN(C)C)=O)C3)C2)=O)c[nH]nc1S(N)(=O)=O C(=O)(CCCC(N)=O)N1C(CCCNC(c2ccc(C)s2)=O)CCC1 CCC1=C(C(=O)NC2CC(CNC(c3ccn4ccnc4c3)=O)C2)SCCO1 c1(C(=O)NC2CN(C(CN(CCC)C)=O)C(C)(C)C2)c(F)ccc(OCC)c1N c1(C(N2C(C(=O)NC(C3CCOC3)C#C)CC3CC32)=O)ncnc(C)c1C c1(OC)cnc(C(N2CC(CNC(=O)CC3CCCN3C)C3(CC3)C2)=O)c(F)c1 N1(C(C(CC)(C)COC)=O)CC2COCC2(C(=O)N(C2COC(C)(C)C2)C)C1 N1(C(C(C)O)=O)CCCC(C2CN(C(c3occ4c3CCC4)=O)C2)C1 N1(C(CC(C)F)=O)CCCN(C(C2(C)CCN(Cc3ccccc3)CC2)=O)CC1 C1(C(N(CCCCN(C)C(c2ccncc2N(C)C)=O)C)=O)CCCCNC1=O c1(OC)ccc(Br)c(NCC(N2CCCC3CC23)=O)c1 N1(C(CC2N(Cc3onc(C)n3)CCC2)=O)CCCN(C(=O)OC(C)C)CC1 c1(C(N2CCC(CCNC(CCNCCC)=O)C2)=O)cc(OC)cc2c1CCC2 c1(C(=O)NC23CCC(C2)N(C(C2CC4(CC4)CO2)=O)C3)ccc2[nH]ccc2n1 N#Cc1sc(-c2ccccc2)cc1NC(=O)CCCNC(=O)CN N1(C(c2cnn(CC)n2)=O)CC(NC(=O)CC(C)NC(N)=O)CC(C)C1 N1(C(C2(CC=C)CC2)=O)CCCCC2(CCN(C(=O)C=CS(=O)(=O)CC)C2)C1 O=C(C1=CC(C(F)(F)F)C1)NC(c1ccc(F)cc1)c1cncc(Br)c1 N1(C(C(c2ccc(F)cc2)CC)=O)CC2(CCC(CNC(=O)C=CCF)O2)C1 c1(NC(=O)OC)ccc(-c2ccc(NC(=O)NC3CCC(O)CC3)nc2)cc1 C1(CCC)CN(C(C2(NC(N)=O)CC2)=O)CC1C(=O)NCCCC1(C(N)=O)CC1 Cn1cnc(C=CC(=O)NC2CCC2CNC(=O)CC2CC2(C)C)c1 CC(CNC(=O)C=CC(C)(C)NC(=O)CC1CSC1)C(F)(F)F C1(NC(C=CCCC)=O)CC2CCC1(NC(c1ccc(CS(N)(=O)=O)cc1)=O)C2 C1(NC(CC2CC(OC(C)(C)C)C23CCC3)=O)CC2CCCCCCC12 c1(C(N2CC(C#N)C3(C2)CCC3)=O)cc(Cl)cc2ccccc12 CC(C)CC(CC(=O)NCCN1CC(CF)C1)NC(=O)C1=NOC(C)C1C C(C(C(C)C(C)C)NC(c1ccc(F)c(O)c1)=O)NC(c1cnc(COC)s1)=O C1(NC(C(C)OCC(C)C)=O)CC(O)(CNC(c2ccon2)=O)C1 Cc1ccc(CNC(=O)CSCCNC(C2(C)CCOC2C)=O)cc1F c1(CC(=O)NCC(CC)NC(=O)C(C(C)CC)N(C)C)ccc2nc[nH]c2c1 C(CC(C)C(=O)N(C(C)CNC(c1cnn(-c2ccc(F)cc2)c1N)=O)C)OC c1(NC(C(C)(c2ccccc2)OC)=O)cc(C)cc2ccoc12 CN1CC(NC(=O)NCCOC2CCOCC2)C(C)(C)C1 c1(C(=O)NCC(=C)CCNC(=O)CC2CCC(=O)O2)coc2ccc(Br)cc12 c1(COC)cc(N2CCCC2CNC(C23CCC(C2)OC3)=O)ncn1 Cc1ccc(CCC(=O)N(CCNC(c2csc(C(F)F)n2)=O)C2CC2)o1 c1(C(=O)NC2CN(C(C(C3CCC3)OC)=O)CC(F)C2)cccc2ncnn12 C1(CCC)(NC(C2CC(=O)NC(C)C2)=O)CCN(C(=O)CC2(CO)CC2)CC1 Cc1c[nH]cc(C(=O)NCC2CCC2NC(=O)Cc2c(F)cccc2F)c1=O c1(C(=O)NC(CC=C)CNC(=O)CC(CC)C2CC2)nnc(O)c(Br)c1O N1(C(C2CCC(N(C)C)C2)=O)CCN(C(=O)CNS(C)(=O)=O)CC1CO c1(CNC(C(N(C(C(CC)SC)=O)C)C2CC2)=O)cc(OC)nn1C c1(C(N2CCN(C(C3ON=C(C)C3)=O)C(CCO)C2)=O)cn2cc(C)ccc2n1 N1(C(c2[nH]cc(C)c2)=O)CCCC(CC(=O)NC(c2nncs2)C)C1 C1(NC(c2n(C(C)C)ccn2)=O)CC=C(C(=O)N2CC(C)C(C)C2C)C1 Cc1c(NC2CCOC(C)C2)ncnc1N(C)C.c12ccnc(n1)S2 C1(C(=O)NCCc2cc[nH]n2)CC2(CCN1C(c1cc(CO)[nH]n1)=O)CC2 C(=O)(CC(C)CC(F)(F)F)NC1C(N(C(C=CC=CC)=O)C)CCCC1 C#CC1(C(N2CCC(NC(C3CCCN3C(=O)C(C)(C)C)=O)CC2)=O)CCCC1 N1(C(C2CC(F)C(=O)N2)=O)CCC(NC(C2(Cc3ccccc3)CC2)=O)C(O)C1 C(=O)(C(CCN(C)C)NC(C1COCC1C(N)=O)=O)NCC1CC(N(C)C)C1 C1(CN(C(c2nc(COCC)sc2)=O)C)CCCN(C(=O)CCC2CC2(Cl)Cl)C1 N1(C(c2ccn(CC(F)F)n2)=O)CC2(CCN2C(=O)CCc2ccc(O)nc2)C1 N1(C(C(=O)NCCCSC)CCc2ccc(Cl)cc2)CC(C)(C)C(O)C(C)(C)C1 Cc1nn(C)c2c(NCC(F)(F)Br)nc(=NC3CCCc4ccc(Br)cc43)[nH]c12 Cc1nccc(-n2cc(C(N3CCCC3CNC3CCCN(C)C3)=O)nn2)c1Cl c1(C(=O)Nc2cnc(CC3CC3)nc2)c[nH]c2c(F)cc(Br)cc2c1=O c1(C(c2n(CC)nnn2)Nc2ccc(C)c(C(=O)OC)c2)ccc([N+](=O)[O-])cc1 N1(C(CCNC(=O)NCC)=O)CCC(CNC(=O)CCCCCOC)C12CC2 N1(C(CCc2cc(C)on2)=O)CCC2CCN(C(=O)Cc3sc(C)nc3C)CC12 C1(CNC(CSCCC)=O)CC2CC(C1)N(C(c1n[nH]cc1Cl)=O)C2 C1(C)(CC)C=C(C(=O)N2CC(NC(=O)CC3NC(=O)NC3=O)C2)C1 CC1=NS(=O)(=O)NC(C)=C1CCC(=O)NCC(C)(C)CNC(=O)Cc1csnn1 c1(N(C)C(C2CNCCOC2)=O)ccc(NC(=O)NC2CCC3CCC23)cc1Cl c1(NC(CC)CC(C)C)ncnc(NCCc2ccccc2F)c1C C1(O)(CCNC(c2n(CC=C)ccc2)=O)CCN(C(C2NC(=O)OC2C)=O)CC1 N1(CC(=O)NC2CC(O)(CNC(C(c3ccn(C)n3)(C)C)=O)C2)C(=O)CCC1=O CC1(C)OCCC1n1nc(C2CSC2)nc1-c1cnn(Cc2ccccn2)c1 C(=O)(CC(C)P(C)(C)=O)NCC(COC)NC(C1CCN(CC(F)(F)F)C1)=O CC(C)(CO)C(CO)NC(=O)C(Cc1cccnc1)NC(=O)C1CC1 c1(C(N2CCCC(CCNC(C(CCOC)C)=O)C2)=O)c2ccccc2nn1C C1(CC(=O)NCC(N2CCSCC2)C)(CC)CCOCC1 N1(CCNC(c2cc(C(C)=O)on2)=O)CCN(C(c2ccn(C)c2C)=O)CC1 c1(C(=O)NC(C2(O)CN(C(=O)CCc3cnc(C4CC4)o3)C2)C)cn(C)c(O)n1 N1(CCC)CCC(N=c2[nH]c(=NC)[nH]c(=NCC3CCCOC3C(C)C)[nH]2)CC1 C(=O)(C1=CC(O)CCC1)N1CCC(OCCNC(Cc2c(C(C)C)con2)=O)C1 c1(C(=O)NCC2C(C)CCN2C(=O)Cc2ccns2)ccc2c(c1)CCCCS2 N1(C(c2cc(CC)sn2)=O)CC2C=CC1C(C(N1CCCC3COCC13)=O)C2 C#CCCN=C(NCC(F)=C(C)C)NCc1cc(Cl)ccc1Br Cc1ccc(N2CC(C(=O)N(CC(O)CNC(=O)CSC(F)F)C)CC2=O)cc1 N1(C(COC(C)C)=O)CCCCC1C(C)NC(=O)Cn1ccnc1 CC(C)CCC(F)C(=O)N1CC2CCCC2(NC(=O)CSC2CCCCO2)C1 C=CC(C(F)(F)F)NC(=O)C(CC=CC)NC(c1[nH]cc(C)c1C)=O C1(C(=O)NC2(CN(C(C3CC(C(F)(F)F)(OC)C3)=O)C)CC2)OC2CCC1CC2 c1(COC)nc(N2CCCC(N(C)C)CC2)cc(N2CCC(C(F)(F)F)CC2)n1 CC(C)C(CCN(C)C(c1scnc1C(F)(F)F)=O)NC(=O)CCC(=O)N(C)C C1(CC(=O)N(CC(CCC)O)C)CN(C(=O)C(O)CCSC)C(C)(C)C1 c1(CNC(C2CN(C(C3N(C(C)=O)CC3)=O)C2)=O)[nH]c(-c2cccnc2)nc1C CC(C(=O)NCC1(CNC(c2ccco2)=O)CC1)(C(F)F)c1ccccc1 c1(C(=O)NC2CCC(NC(c3c(N(C)C)cccc3)=O)CC2)cc2c(s1)CCC2 c1(-c2scc(CC(=O)NC3(CCNC(C4CCOC4)=O)CC3)n2)ccccc1F N1(C(=O)CCn2cncn2)CCC2CC12C(N1CCCC(CCF)C1)=O c1(-c2ccn(C)n2)ccccc1C(N1CCC(F)(c2cn(CCN(C)C)nn2)C1)=O Cn1c(SCCCO)nnc1-c1c[nH]nc1O C(=O)(CC(O)CCSC)N(CCC)CCNC(c1nc(OC)c(C)s1)=O N1(CC(=O)NCCN(C(C2CN3CCC2CC3)=O)CC)C(=O)CC(C)(C)C1=O C#Cc1ccc(CC(=O)N(C(CC)C(=O)OC)C(CC)=NC(=O)NCC(C)(COC)CC)cc1 C(=O)(CC(C)(C)N(C)C)N(C1CCN(C(=O)CCc2ccccc2)C1)C N1(C(c2nn(CC)c(=O)cc2)=O)CC2CCN(C(C3CC(C)(F)C3)=O)C2C1 c1(CCC)n[nH]c(=NCC(CC(C)C)NC(C23CC4CC(C2)CC(C)(C4)C3)=O)o1 Cc1c(NC(C2CC(O)(C(F)(F)F)C2)=O)cccc1N1C(=O)CCC1=O C1(C(=O)NC23CCCC2N(c2ncc(Br)cn2)CC3)CNc2ccccc2O1 N1(C(C2CCN(S(C)(=O)=O)CC2)=O)CC2CCC(C1)N2C(C1CN(C(N)=O)C1)=O N1(C(C(CC)NC(N)=O)=O)CC2(C1)SCCC2NC(=O)CC1=CCOCC1 CN1CCN(C(=O)CCC(=O)N2CCCC2)CC1CNC(=O)Cn1ncnn1 N1(C(c2nc(C(N)=O)sc2)=O)CCC2(CC1)CC2CNC(=O)C=CC1CC1 N12C3CCC1CN(C3)C(=O)C1C(CC=CC1)C2=O.c1(COC)cccc(B(O)O)c1 c1(C(=O)NC(CCCNC(C2C(C)CC2)=O)C)ccc(Cl)c(O)c1 C(=O)(C(F)(F)CCn1ccnn1)N1CC2C(CNC(=O)COC3COC3)C2C1 c1(OC)cccc(C(=O)NC2CCC2NC(=O)C(c2ccc(C)cc2)O)c1OC C1(C(=O)NCc2ccc(O)cc2F)C(C2CC2)CCN1C(=O)CCOC1CC1 C1(CCOCC)CCCN(c2cc(N3CCC(C)=C(Br)C3)nc(CC)n2)CC1 N1(C(C2(OC)CCN(C(c3nc[nH]n3)=O)C2)=O)CCC(C)C(F)(F)C1 N1(C(C2CC(=O)C2)=O)CC(F)(CNC(=O)CCn2cncn2)C1 c1(C(=O)NC23CC2CN(C(=O)C(F)CC2CCCC2)C3)cnc2n1CCS2 c1(C(N2C(CC(=O)NC(CCC)CO)CCC2)=O)nc(C)oc1C c1(C2C(C(=O)NCC3(CNC(C(C)SC)=O)CCC3)C2)ccnn1C N1(C(C2(C(=O)NC)CC2)=O)CCCC2CN(c3ccc(S(C)(=O)=O)cn3)CCC12 Cc1ccnc(C(N2CCCC(C(F)(F)F)(CNC(C3(CO)CC3)=O)C2)=O)c1N N(C1CN(C(c2c(C)[nH][nH]c2=N)=O)CCc2ccccc21)C(C(CSC)(C)C)=O c1(CN2CCCC(C(=O)Nc3cc(CCC)no3)CC2)ccc([N+](=O)[O-])c(F)c1 C1(Nc2ccc(C)c(N3CCCS3(=O)=O)c2)COc2cc(Cl)ccc2C1 N1(C(CN(C2CCC2)C(c2ccccn2)=O)=O)CCOCC1Cc1cccc(O)c1 N1(C(C2(F)CCN(C(C3(C)CC=CC3)=O)CC2)=O)CCCC2(CC1)CC2 c1(-c2c(SC)nc(Cl)nc2N)ccc2c(c1)CN(C)C2=O C(CCCC(C)(C)NC(C1C=CC(C(=O)NC)C1)=O)NC(C=C(COC)C)=O CC1CC2(CC(C(N3CCCC3CNC(c3ccc([N+](=O)[O-])o3)=O)=O)C2)C1 C=CC1(C(=O)Nc2cc(C)c(O)c(C)c2)CCN(C(C2CC23CC3)=O)CC1 N1(C(C2(C(=O)NC)CC2)=O)CC2(CC(NC(c3ncccc3O)=O)C2)C1 N1(Cc2cccc(OC)n2)CCC2(CC1)CC2C(=O)NCC(=O)NCC(C)C c1(NC(=O)NC2C(C)N(CCO)CC2)ccc(Cl)cc1NC(c1ccccc1)=O C(=O)(CC1COc2ccccc21)NCC(C1(O)CN(C(CC=C(C)C)=O)C1)(C)C c1(SC)ccccc1C(C(=O)O)NC(=O)C(CO)c1ccccc1 c1(C(N2CCC(NC(CCCCC)=O)C2)=O)ccc(C)c(C(C)=O)c1 C1(NC(c2[nH]cc(C)c2)=O)CC2(C1)CC2NC(c1ccccc1CCN(C)C)=O c1(SC)nc(C(=O)NCC#CCNC(=O)Cc2cc(C)on2)cs1 c1(NCC2(CC(C)C)CCC2)cc(N(C)Cc2nncs2)ncn1 C(=O)(CCN(OC)C(=O)C1(C)CCN1C(=O)COCCCN(C)C)OC C(C(C)(C(C)C)NC(=O)C(C)CN1CCCCC1)NC(CC1CC(SC)C1)=O c1(OC)cc(C(=O)NCC2CCCCN2C(C2CN(C(C)=O)C2)=O)ccc1C#N Cn1ccc(CCC(=O)NC(C2CCOC2)CNC(=O)Cn2cccn2)n1 C1(c2ccncc2F)(CNCCc2ccccn2)CCNCC1 C1(C)(NC(COCCC=C)=O)CCN(C(C2CCC(COC)O2)=O)CC1 N1(C(c2[nH]c(=NCC)sc2)=O)CCC2(NC(=O)C=CC=C(Cl)Cl)CCCC12 Cc1ccc(C(=O)NC2COCC2NC(=O)CCc2ncccc2C)c(F)c1 N(C(=NCCOC1CCOC1)N1CCN(CC(N)=O)C(=O)C1)C(CC(F)(F)F)C N1(C(c2c(C)noc2)=O)CCN2CCN(C(=O)C(F)CCC(C)(C)C)CC2C1 c12ccc(cc1)[nH]c2=O.C1(CCC(=O)N(C(C)=O)C2CC2)CCC(C)O1 c1(CC)cccc(NC(=O)CC(CNC(c2cnn(C(F)F)c2)=O)OC)c1C c1(C(=O)NC2C(CNC(C3(CC#C)CC3)=O)COC2)cc[nH]c(=N)n1 Cc1ccnnc1C(=O)NC1CC(CNC(=O)C(F)(F)c2csc(Cl)c2)C1 Cc1cc(=NCC(C)C2CC2)[nH]c(=NCCc2cnc3n2CCOC3)[nH]1 C1(NC(Cc2cncc(C)c2)=O)CCN(C(C2CN(C(=O)N(C)C)C2)=O)C12CCC2 N1(C(C2CN(C)C2)=O)CCCC2(NC(=O)COC3CCC(F)(F)CC3)CCCC12 Cc1ccc(OCC(N2CC3C(C2)N3C(=O)CN2CCCCC2=O)=O)cc1 C12(NC(C(CC)c3ccccc3)=O)CCCC1N(Cc1ccc(I)cc1)CC2 C1(NC(C2CC(SC)C2)=O)CCC2(CC1)CN(C(=O)CC1C=CCC1)CCO2 C#CCC(C)(C(=O)NC(CO)CC#CC)NC(=O)COC1(C)CCC1 c1(C(N2CCCC(CN(C(COC)=O)C)C2)=O)cccc2c(C3CCC3)c[nH]c12 C1(NC(c2cc(C3CCCC3)no2)=O)CCSC12CN(C(C1CCS1(=O)=O)=O)C2 c1(C(C)C)cccc(C(N2CCC(NC(C3(C(C)(C)O)CC3)=O)CC2)=O)c1 Cn1cc(C(=O)NC2CCCCCN(C(=O)C=C3CC3)C2)c(=O)c(Br)c1 c1(C(=O)NC2CC2(F)F)ccc(-c2cnn(CCN3CCCC3)c2)s1 Cc1cccc(C)c1CNC(C1(C(C)NC(=O)C=Cc2cncn2C)CC1)=O CC(C)C(CN(CCCO)C(=O)NCc1cccc(C2CCC2)c1)C(C)C N1(C(Cn2cc(C(=O)NC)nn2)=O)CCCC(NC(c2ccc(C)c(O)n2)=O)C1C CCC(Cc1ccccc1Br)C(=O)NCC1(O)CC(C)(C)C1 Cc1cnc(F)c(C(=O)NC2CC(C)N(C(C3CN(C4CCOC4)C3)=O)C2)c1 CN1CCCC(C)(C(=O)NC2CC3CC2N(C(=O)CN=S(C)(C)=O)C3)C1 N1(C(c2cncc(CNC(CC3CCC(C)C3)=O)c2)=O)CC2CCC(C1)C2O C1(CC(=O)NCC2CC(NC(=O)C=C3CCCCC3)C2)CCC12CCC2 c1(C(N(C(C)CCNC(c2cnnn2C2CC2)=O)C)=O)ccn2nccc2c1 c1(C(CC)C)ccc(C(=O)N(CCNC(=O)C(C)(COC)OC)CC)cc1 C(=O)(CCS(C)(=O)=O)NC(C1CCN(C(=O)CC2CCCOCC2)C1)C c1(C(N(CC(CC)NC(C2CC(C(C)C)C2)=O)C)=O)cccnc1CO C1(CNC(c2c(Cl)cnc(C)n2)=O)CC2CCC(C1)N2S(=O)(=O)c1ccc(Br)s1 c1(C(N2CCCN(C(C(CC)F)=O)CC2C)=O)ccc(F)c(S(C)(=O)=O)c1 C1(C(=O)NCCC(=C)CNC(=O)C(C)(C(C)C)OC)CCc2c(n[nH]c2C)C1 N1(C(c2c(CC)csc2)=O)CCN(C(=O)COC2CCOCC2)C(COC)C1 C#CC1CCCN(C(c2ccc(C(F)F)cc2C)C(=O)NCCC#N)C1 c1(OCC(=O)NC2C3N(C(CC(C)OC)=O)C(CC3)C2)ccc2ccccc2c1 C=CCCC(C(=O)NCc1cc(C)c(CC)o1)NC(=O)CC1CC(C2CC2)C1 Cc1cc(C(N2CCN(C(=O)CCC(F)(F)F)CC23CC3)=O)c(F)cc1Br Cc1ccc(CO)c(NC(=O)C(CNC(=O)CN(C)C(N)=O)N(C)C)c1 C12(CNC(Cn3c(C)cc(C)n3)=O)CN(C(=O)CN=S(C)(C)=O)CC(F)(C1)C2 C(=O)(CS(=O)(=O)C(C)C)NCC1(OC)CCN(C(=O)C(C2CCOCC2)C)CC1 CC1(CNC(=O)Cc2cnns2)CCCN1C(c1cccn1C1CCCC1)=O C12(C(=O)NCCCCC3CN(C(c4sccc4CO)=O)C3)CCCC1OCC2 CS(=O)(=O)CCCC(=O)NCC1CN(C(=O)Cc2ccccc2Cl)CC12CC2 C1(CNC(CSCC(C)C)=O)(CO)CCN(C(=O)CCOC2CC2)C1 N1(C(c2n(CC)ncc2)=O)CCC2(CC1)CC2C(=O)NC(c1ncccn1)CC C(CC(C)(C)C)(C(=O)N1CC2CC(CNC(c3ccc(N)c(Cl)c3)=O)C2C1)OC C1(C#N)(C(=O)NCC(C(=O)NCc2n(CCC)ccn2)OC)CC(C)C1 c1(C(N(CCNC(C2CCC3C2C3(F)F)=O)CC)=O)coc2c(Br)cccc12 c1(C(C(=O)NCC(C)CNC(c2ccc(F)o2)=O)(F)F)cccc(Br)n1 c1(N2CCC(O)(C(C)NC(=O)C(C)(C)N(C)C)C2)ncnc2ccsc12 CC(C)C(O)C(F)(F)C(=O)NCC1C(Cn2cc(-c3cccc(=O)o3)nn2)C1(F)F N1(C(CC(C)C(F)F)=O)CCC(C2CCCN(C(C3CC34CC4)=O)C2)C1 c1(C2C(Cc3nc(CS(=O)(=O)Cc4nc[nH]n4)on3)C2)cccc(F)c1 C(C(C(=O)NCCN1CCCOCC1)C(C)(C)C)NC(c1c(C)scc1)=O C(=O)(C(C)C(=O)N1CCOCC1CNCc1nc(-c2ccc(Cl)cc2)no1)OC C1(CC)C(CC(=O)NCCN(C)C(C2CCC2c2nc(S)n[nH]2)=O)C1(F)F O=C1CCC(C(=O)NC2C=CC(C(=O)Nc3ccccc3C(F)(F)F)C2)=NN1 c1(CCCN)nc(C(C)C)no1.C1(C(OCC)OCC)CCOCC1 c1(CC(=O)NC2CN(C(c3c(COC)ncs3)=O)CC2O)cc(Br)ccc1C c1(C(C)=O)cn(C)nc1C(=O)NCC(C(C)(C)C)NC(=O)CCCCOC(C)C Cn1cc(Cl)cc1C(=O)NCCCOCCNC(c1ccnnc1NCCO)=O CCC(C)C(CC(=O)N(C1CSC1)CC)NC(c1coc(C)n1)=O N1(C(C(C)N2CCC2)=O)CCCCC1C1CCCN(C(c2ccc(C3CC3)s2)=O)C1 C(=O)(CCC1=NNC(=O)CC1)NCC12C(CN(C(C(=O)NCC)=O)C1)CC2 N1(C(CCNC(=O)OCC)=O)CCC(NC(C2(C)CCN(C)C2)=O)CC1C c1(C(=O)NCC2CCCCN(C(C3CC(OC)C3)=O)C2)cn2ccccc2n1 C1(NC(CCCOCC=C)=O)CCC(CC(=O)NCCNC(=O)CO)CC1 c1(OC)cc(C(C)NCc2ccc(F)nc2F)ccc1OCC(C)C N1(C(CCc2c(C)n(C)nc2)=O)CCCCC(NC(=O)C(C)(C)CO)C1 C1(NC(CCCC#C)=O)CCOC2(CCN(c3cc(S(C)(=O)=O)ncn3)CC2)C1 C(=O)(C(C)S(N)(=O)=O)NC(CC)CN(C)C(C1CCS(=O)CC1)=O c1(OC)cc(C(N2CC(CNC(=O)Cc3cnco3)CC2C)=O)cc([N+](=O)[O-])c1 c1(C(N2CC3C(CNC(C4(CC)CC4(F)F)=O)C3C2)=O)cc(C)c(F)cc1F C1(CC)(NC(c2cccn(C)c2=O)=O)CCN(C(=O)C(F)C2CCOC2)CC1 N1(C(=O)CCc2cnc(O)[nH]2)CCN(C(=O)CCCc2cccs2)C2COCC12 C(=O)(C(F)C(F)(F)C(F)(F)F)NC(=O)CC1(c2cn(CCC(C)C)nn2)CCC1 C12(NC(C3CC(=C)C3)=O)CCN(C(=O)CCCc3csc(=N)[nH]3)CCC1C2 CC1(C)CCC=C(C(=O)NCCOC2CN(C(c3cccc4c3OCC4)=O)C2)C1 N1(C(CN(c2ccsc2)C)=O)CCC(NC(=O)C=C2CCC2)CC(C)(C)C1 C(=O)(C(CNC(C1CCCC1O)=O)CC(C)C)NCCC(=O)NC(CC)C c1(C(=O)NCC2C3CCCC2N(C(c2ccc[nH]2)=O)C3)nccc2cccnc12 c1(CNC(c2nnnn2Cc2cccs2)(COC)C)cnn(C)c1 c1(OC)c(C(=O)NCCC2CN(C(c3ccon3)=O)CC2C)ccnc1Cl c1(OC)cnc(CNC(=O)CCC2CCCN(C(c3cc(OC)cs3)=O)C2)cn1 N1(C(c2ccc(OC)nc2C)C(=O)NC2CC2)CCc2cc(C)c([N+](=O)[O-])cc21 C12(CNC(C3(CC=C)CCOC3)=O)CCC(CN(C(=O)CCC(CC)CC)C1)C2 c1(C(=O)NC2CC(C)N(C(C3(C4CCC4)CC3)=O)C2)c([N+](=O)[O-])cnn1C CC1(C)C(CNC(=O)CSC2CC2)CCN1C(c1ccsc1Br)=O c1(C(N(CCNC(C2C(CC)C2)=O)CCOCCO)=O)ccc(Br)c(C)c1 c1(C(N2C(CCNC(=O)CC3CSCCS3)CCC2)=O)cc(F)cc2nc[nH]c12 CC1(C)CN(C(C2(C#N)CCC2)=O)CC(CNC(c2cncc3nc[nH]c23)=O)O1 C1(NC(c2cncc(Cl)c2)=O)CCCCN(C(C2(CCF)CCOCC2)=O)C1 OC1CCC(c2nnnn2C2CCOCC2)(Nc2cnccc2SCCF)CC1 CCCC(C)CC(=O)NC(C)Cn1cc(-c2cccc(F)c2)nn1 N12CC3CC1CC3NCC2=O.c1(C(C)C)cc(C(=O)N)ccn1.C1(C=O)CCCC1 C(=O)(C(C)CC(=O)N1CCOC(C2(On3cccn3)CC2)C1)OC Cn1cc(NCc2ccc(I)cc2)cc1C(=O)NCC(c1ccc(F)cc1)O C1(F)(CNC(=O)C=CCn2cncn2)CCN(C(c2ncccc2C2CC2)=O)C1 C(=O)(C1=C(C)CCCC1)N1CCC(NC(C2(SCC)CC2)=O)C(C)C1 C(C1=COCCC1)(c1n(CCOC)nnn1)NCCN(C1CCC1)C c1(N(C)C)ccc(F)c(C(N2CCC(NC(C3CCC(C)(C)O3)=O)C2)=O)c1 C(C(C)(C)C(C)(C)C)NC(C(C)N(C(=O)CN1CC(C)(OC)C1)CC)=O N1(c2nc(C)nc(O)c2)Cc2nccn2CC(NC(c2ccc(Cl)s2)=O)C1 C(=O)(C(F)(F)C(F)F)NC1(C)CC(NC(c2ccc(-c3ccccn3)s2)=O)C1 C(C(C)CC(=O)NC(C1CN(C(C2CCC(C)C2)=O)CCO1)C)OC O=C1CC(C2CC2)NC(=O)C2(CCC2)N1.c1(C2C(SC)C2)cncs1 C12(NC(C=CC=CC)=O)CCCC1(F)CN(C(C1(C#N)CCSCC1)=O)C2 C=CC(C)(O)C(=O)NCC1C(C)CCN1C(=O)CC1CC=CCC1 c1(NC(C(C(=O)OC)C)C=O)ccc2c(c1)OCCC2 C1(CNC(c2c(C)n(C)nc2)=O)CC(F)(F)CN1C(c1ccc(C(C)C)cn1)=O C1(NC(C(C)N(C(C2(C#C)CC2)=O)C2CC2)=O)CC(=O)N(O)C1 c1(NC(C(=O)NCC2(NS(C)(=O)=O)CCSC2)=O)ccc(Br)c2c1OCCO2 C1(NC(C2OCCN(C(CC(C)=C(C)C)=O)C2)=O)CCCCCC1(C)C Nc1c(F)c(C(N2CC=CC(NC(C3CCCC(F)(F)C3)=O)C2)=O)cc(F)c1F C1(NC(CC(C)n2cccn2)=O)CC2CCC1N2C(=O)C(c1ccccc1)C c1(C(=O)NCC23CC(CNC(CCCC=C)=O)(OC2)C3)ccc(C(C)C)nc1O C12(C(N(CCN(C(c3c[nH]ccc3=O)=O)CC)CC)=O)C3CCC(CC13)C2(F)F c1(C(=O)NC2CN(C(C3(CC=C)CCOC3)=O)CC2CC)ccc2sncc2c1 Nc1cc(Br)ccc1CNCc1ccc(F)cc1 c1(OC)cc(C)c(-c2ccc(NCc3cc(Br)ccc3C(F)(F)F)c(F)c2)cn1 CCCC(CCC)C(=O)N1CCC(NC(=O)CCc2nncn2C)C1CC C12(C(=O)NC3CCC(CNC(=O)CC4COCCO4)C3)CCCN(CC1)C2 O=C(CCCCc1cccs1)NNC(=O)NC1CCCC1 CCCC(C(=O)N1CC(C2CN(C(=O)CC3(O)CCOC3)C2)C1)C(C)C N1(C(c2cc(CCC)[nH]n2)=O)CC(NC(=O)CCP(C)(C)=O)CCC1C N1(C(c2ccn(CCCC)n2)=O)CC(CNC(c2cnns2)=O)C(F)(F)C1 Cc1cc2[nH]c(=O)c(C(=O)NCC(C(C)C)NC(C3CCOC3)=O)cn2n1 c1(NC)ccc(C(=O)NCCCOCCC(=O)NC(C)C(C)(C)CO)nc1 CCC(C)(CC(=O)NC1CCC1CNC(=O)C=Cc1nccs1)C(=O)OC c1(C(=O)NC(C(C)OC)C)c(C)sc(C)c1Br C1(NC(C2(Br)C(C)(C)C2)=O)(CO)CCCN(C(=O)CCC2CCC2)C1 C(=O)(CC(C)C(F)F)NC(CNC(CC1CCN(C(C)C)CC1)=O)C(C)(C)C C=CCCCCCC(=O)NCC1CC1NC(c1ccc[nH]1)=O CC(C)C(C(=O)NCCN(C1CCCC1)C(=O)C=Cc1ccc(Cl)s1)NC(N)=O C12(NC(C3CC3c3cn[nH]c3)=O)CC1CN(C(C1CCCCO1)=O)C2 N1(c2snc(C(=O)OC)n2)CC2CC1CN(C(=O)COC1CCOC1)C2 Cc1oc(C(C)C)cc1C(=O)NCc1cn(C(Cc2ccccc2)C(N)=O)nn1 N1(C(CN(C(=O)CCSCC(N)=O)CC)=O)CCCC(CF)C1 C1(NC(c2cnc(OCC)s2)=O)CCC(C)N(C(=O)CCc2ccc(F)cc2)C1 N1(C(CCCC(CCC)C)=O)CC2CCC1C1CN(C(=O)C(C)N3CCC3)CC21 C1(CC(NC(=NC)NCC(C)(C)C(F)F)C#C)CCc2ccccc2C1 C(=O)(C(C)C(O)C(C)C)NCCC1CCN(C(Cc2c(OC)ccc(C)c2)=O)C1 C(=O)(C1=NOC(C)C1)NCCC1CCN(C(C(COC)NC(C)=O)=O)CC1 c1(CNC(C(n2cc(-c3c(Cl)cncc3Cl)nn2)C)=O)nnc2n1CCC2 C(CC(C(C)(C)C)NC(C1COCC1(C)C)=O)N(C)C(c1cc(Cl)n(C)n1)=O c1(C(=O)NCCCn2ccnc2)ccc(-c2cn(Cc3ccccc3)nn2)cc1 c1(OC)ccc2[nH]c(C(N3CCN(CC(=O)O)CC3(C)C)=O)cc2c1Cl CN1CCC(NC(=O)C(COC(C)(C)C)n2cc(-c3cscn3)nn2)C(C)(C)C1 C1(C(=O)OC(C)(C)C)CCCCN(C(c2cccc(-c3cn(C)nn3)c2)=O)C1=O c1(C(=O)NCCN(CCC)C(C2(OC)CCC2)=O)cc(Cl)cc(Cl)c1OC C1(N(C)C(c2cnc(C3CC3)o2)=O)CN(C(=O)C=CCOC(C)(C)C)CC1O CC(C)C(CNC(=O)C(=O)Nc1noc(CNC(C)(C)C)n1)Sc1ccccc1 C=CC1CN(C(CC(c2cccs2)NC(N)=O)=O)CCO1 n1(C(C(=O)OCC)C)cc(CN(C)Cc2ccc(Cl)o2)nn1 C1(C(=O)NCC(CC(C)C)NC(c2cc[nH]n2)=O)CC2COCC2C1 C#CC1CN(C(=O)C(CC=C)NC(=O)C(C)Cn2cccn2)CCO1 c1(C(=O)NC2CC(C)(C)N(C(c3cnncc3O)=O)C2)ccn2nnnc2c1 N1(C(c2c(CC)nn[nH]2)=O)CCC2(CC1)CCN(C(C1(C)CCN(C)C1)=O)CC2 C1(C(N(C)CC2(O)CN(C(=O)C(=O)NC3CC3)C2)=O)CCC(F)(F)CC1(C)C N1(C(C(C)OC2CCCCCC2)=O)CC(NC(=O)CCC(C)(C)C)C2(CC2)C1 CC(C)CC(C(=O)NCc1ncoc1C(C)C)NC(=O)Cc1ccccc1O c1(C(=O)NC(CNC(C(CCC)C)=O)C(C)C)cc(Br)c2c(c1)nnn2C C(=O)(C1=CC2CCC1C2)NCCCC(C)(C)NC(CCN(CC(F)(F)F)C)=O c1(N(C)CC)ccc(C(=O)NCCC2(NC(=O)CC3(O)CCC3)CCC2)cc1 c1(C(N2CCC(C(C)CNC(C3CC3(C)C)=O)CC2)=O)ccc([N+](=O)[O-])cc1Cl CP(C)(=O)CC(=O)NC(CCC1CC1)C(=O)N1CC(OC(F)F)C1 C1(OC)(CNC(c2oc(-c3cnn(C)c3)nc2C)=O)CCN(C(C2CC2C)=O)C1 C(=O)(C1=CC2CCCCCC12)NCCC(C)(C)NC(COCCN(C)C)=O N1(C(C2CC(n3cc(CNC=O)nn3)C2)=O)CC2COCC(C2)C1 Cc1oc2ccccc2c1C(N1CCC(C(=O)NCC2(CNC3CC3)CC2)C1)=O C1(C(C)(C)C)C(=O)NCCNC(=O)C2(CC2)C(=O)N1C.C1(O)(CC2CCC2)CCC1 c1(NCCCC(=C)C)ccc(S(=O)(=O)NCCn2ccnc2)cc1F c1(N2CC(OC)OC(C)(C)C2)cc2cc(Br)ccc2nc1Cl CC(C)(C(=O)NCCC(C=O)NC(=O)CC1CCN(CC(F)(F)F)C1)C(F)(F)F c1(C(=O)NC(CN(C(COCCC)=O)CC)CC)oc2ccc(Cl)cc2c1C N1(C(Cc2nc(C)on2)=O)CC2(CCCN2C(c2cnc(OCF)cn2)=O)C1 S(=O)(=O)(c1c(F)cc(C)cc1Br)NC1C(OCCOC)COCC1 CC1(C(=O)NCC2CC3C=CC2C3)CCN(C(c2cnc(O)o2)=O)CC1 C1(NC(C2(CCCC)CCC2)=O)CC2CC1CN(C(c1ncnn1CC)=O)C2 C1(NC(c2n[nH]cc2[N+](=O)[O-])=O)CC2CC(NC(C3CCCS3(=O)=O)=O)CC12 C(C(CCC)C(=O)NC(N1CCC(O)C1)(C)C)NC(CCOCC#C)=O C(CCC(=O)N(C)CC1CCCN1C(=O)Cn1cnc(C(F)(F)F)c1)OC n1(CC)ccnc1CN(C(=O)C(C)(C)C1CCN(C(=O)C(C)NC=O)C1)C Cn1ccc(C(N2CCC(CC(=O)NCCc3ccc(Br)s3)C2)=O)c1CC(=O)O C=CC1(C(=O)NCCC(=O)NCCNC(=O)C(C)C)CCOCC1 C1(NC(c2cn(CC(CC)O)nn2)=O)CC2CC1CN(C(=O)C=CC1CC1)C2 C(C)(CCC(=O)NCC1(C(=O)N(c2cccc(Cl)c2)C)CCCC1)SC c1(OC)ccccc1CC(N1CC(N(C)C(C2CCSC2)=O)C1)=O N1(Cc2c(C)nn(CCO)c2)CCN(C)C(c2cccs2)C1 C1(CNC(C2(CC#C)CCC2)=O)CC2(CC2)CN1C(=O)Cc1ccc(C#N)nc1 c1(C(=O)NCC2C(NC(c3ccncc3CN)=O)CCC2)c(F)ccc(F)c1F N1(C(CNC(c2cccc(C)c2F)=O)=O)CC2C3CCC(C2C1)N(C(=O)CO)C3 C12(C(=O)NC(C=C)CO)CCN(C(=O)CNC(N)=O)CCC1C2 C#Cc1cc(C(=O)NCC(C)(CC)NC(c2ccc(C)c(C)c2)=O)ccc1C C1(CC)CC(CC(=O)NC2CC(C(F)F)(NC(=O)CCn3ccnc3)C2)CCO1 N1(C(c2cccc(SC)c2)C(=O)NC(CC)C)CCC(OC)C(OC)C1 N1(C(COC(CC)(C)C)=O)CC2CCN(C(C3CC(O)(C(F)(F)F)C3)=O)C2C1 C(=O)(C1CCCn2nccc21)N1CCC(=CCNC(c2csnn2)=O)CC1 C12(CNC(c3csc(O)n3)=O)CCCCC1CN(C(c1ccc(CO)o1)=O)C2 N1(C(c2c(OC(C)C)n[nH]c2)=O)CCC2(CCN(C(=O)C(C)C(F)(F)F)C2)C1 O(NC(=O)C(C)OCCNC(C1CN2CCC1C2)=O)CC1CC(=C)C1 C12(NC(COC(CC)(C)C)=O)CC(C1)N(C(=O)C(C)(C)NC1CCCC1)C2 c1(OC(C)C(=O)NCC2CN(C(C3CCCCC3O)=O)CCO2)ccccc1Cl [N-]=[N+]=NCCCCC(=O)N1C2CCC1C(C(N1CCC(O)C(O)C1)=O)C2 Cc1cc(NC(C2CC(O)C2)=O)ccc1NC(c1snc(C)c1Br)=O C(CC(C(=O)NCCN(C1CCCC1)Cc1cn(CC(N)=O)nn1)NC=O)SC C(=O)(CS(=O)(=O)C1CCCC1)NC1CN(C(CCCOC(C)C)=O)CC(F)C1 N1(C(c2c(SC)cnn2C)=O)CC2CCC1CN2C(=O)CNc1ccc(C)cc1 Cc1csc(=O)n1CC(=O)NC1(CF)CCN(C(=O)C(C)N2CCC2)C1 C12(C(=O)NCC(C)SC)CC(CO1)N(C(c1ncc(F)cc1N)=O)C2 Cc1cc(=NC(=O)CN(CC(C)C(F)(F)F)Cc2ccccc2)[nH]o1 C1(N(C(=O)C(F)OC(F)(F)F)C)CCCCN(C(=O)Cc2cc(C(F)(F)F)co2)C1 C1(CC(=O)NC2(CNC(C(C)(C)c3cncs3)=O)CC2)CCCCC1O C=C1CCN(C(=O)C(C)=CC(C)(C)C)C(C(N2CC(COC)C2(C)C)=O)C1 c1(CCCC(=O)NCC2CC(NC(C3(CF)COC3)=O)C2)ccc(C2CC2)cc1 Cc1nn(CC(=O)NC2(C)CCN(C(C3(F)CC=CCC3)=O)C2)c2ncccc12 n1(C(C(=O)N(CCNC(c2ccc(C)c(F)c2)=O)CC)C)cnc2ccccc12 N1(CC2CCC(CCCCC)O2)CCCC(NC(C)=O)C1 c1(C(C(=O)NC2C(NC(c3conc3C3CCC3)=O)CCC2)O)ccc(F)cc1 c1(NC(=O)NCC2(COC)CCOC2)cc(C)cc2c[nH]nc12 Cc1c(S(=O)(=O)N2CCCC(C(=O)NCCc3cnn[nH]3)C2)c2ccccc2n1C C=CCC(C(=O)OC)NC(C1CC(NC(=O)CCN2CCCC2=O)C1)=O N1(C(CCC#C)=O)CCN(C(=O)CC2CCC(OC)CC2)C2CCCC12 C1(C(=O)NCCC(N2C(C)CC(CO)C2)=O)CCC(=O)N(C)C1 C(CCO)(CC(C)C)NC(=O)NCC1(OC)CCCC1 C1(C(N2C(C(C)NC(=O)CCc3cncs3)CCCC2)=O)OCCCC1(C)C N1(C(C2CN(S(=O)(=O)C(F)F)C2)=O)CCN(C(C2CC2F)=O)C(CO)C1 CC1(C)COC(C(N2CCC(NC(=O)CC3CC4C=CC3CC4)C2)=O)CO1 c1(NCC2CCCCN(C(c3ccc(COC)[nH]3)=O)C2)ncccc1[N+](=O)[O-] c1(OC)ccn2c(C(N3CCCCC(NC(C4(C)CSC4)=O)C3)=O)cnc2c1 C123CCC(CC1NC2=O)C3.C1(C(N2C(C)(CCO)CC2)=O)CCCN1C=O N1(C(C2CC(C)(CC)C2)=O)CC(N(C(=O)Cc2cccc(F)c2F)C)C(C)(C)C1 C(N=c1[nH]c2cccnc2s1)C1(O)CCCN(C(C(n2ncc(C)c2)C)=O)C1 Cc1ccc(OCC(=O)NC(CNC(=O)COCC2(F)CC2)CC(C)C)cc1 c1(C(=O)NC2CN(C(C(C)(C)N(C)C)=O)CC23CC3)cccc(S(C)=O)c1 C(=O)(C(C)C(C)(C)C)N(CCC(=O)NC(c1nccn1C)C)C1CC1 CCC(C(=O)OC)C(=O)NC1(C(=O)N(C2CC(SC)C2)C)CCN(C)C1 c1(NC(c2nnnn2CCSC)(C)COC)cccc(C(N(CCCC)C)=O)c1 CC(CC(N)=O)NC(c1cc(CCNC(=O)CC2CSC2)on1)=O N1(C(C2N(C(CCn3ncc(C)c3)=O)CCC2C)=O)CC2(CNC(=O)N2C)C1 c1(-c2cn(CC3N(C(=O)COc4ccccn4)CC=C3)nn2)ccc(CO)cn1 C1(CN(CCCC)C(=O)Cc2cccnc2)CCN(C(=O)C2=CCOC2)CC1 C1(NC(C(c2cnn(C)c2)C)=O)CN(C(=O)C(C)N(C)C)CC1(C)C N1(C(c2n(C(C)C)ncc2Br)=O)CCC2CCC(NC(=O)CC(C)(C)C)C1C2 c1(NC(c2c(C3CN(C(C(OC)OC)=O)C3)ocn2)=O)cc(OC)sc1C C1(C(=O)NCCC(C)CCO)C2CC3C(C2NC(=O)C(c2ccnn2C)C)C13 c1(OC)ncc(C2CC2)cc1CNC1CCCC1Oc1ccccc1 C1(CCNC(c2n(CC#C)ccc2)=O)COCCN1C(=O)CCc1nc(=N)[nH][nH]1 c1(C(N2CC=CC(NC(c3cocc3Br)=O)C2)=O)cc2ccccn2c1 c1(C(=O)NC(C(CO)NC(CC(C)C2CC2)=O)C)cc2sccc2[nH]1 CN(OC1CCCC1)C(=O)CC1(C(C2CC2)NC(c2cc[n+]([O-])cc2)=O)CC1 C1(NC(C2CC2CF)=O)CN(C(c2cc3cccc(Cl)c3s2)=O)CC2(CCC2)C1 CC1=NOC(C(=O)NC(C)CCCNC(C2CC(O)C2)=O)C1 N1(C(c2cc(COC)on2)=O)CCC(N(C(=O)C(C)C(C)C)C)CC1 c1(C(=O)NC(c2cnc[nH]2)C)ccc(-c2cncc(N)c2)cc1 c1(C(N(C2CCCN(C(C3CC(C)C3)=O)C2)CCC)=O)ccc2ccncc2c1 N1(C(CCSCC(C)C)=O)CCN(C(C2OCCOC2C)=O)C(c2ncc[nH]2)C1 N1(C)CC2CC1CN2C(C)=O.C1(C(=O)O)(OC)CC(C(F)(F)F)(OC)C1 C1(CC)(NC(=O)CC(C)CNC(=O)C=Cc2cnccn2)CCCCCC1 N1(C(CCC(C)OCC)=O)CC2(CCN2C(=O)CC(C(C)C)c2ccccc2)C1 C1(C(=O)NC2(CC=C)CCCN(C(=O)C(OC)OC)C2)CCc2ccnn2C1 c1(NC(C2N(C(C(C)OCC=C)=O)CC(O)C2)=O)cncc(Br)c1C c1(C(=O)NC(C2CCOC2)CNC(C2CC(OC)C2)=O)coc(Br)n1 N1(C(c2cn(CCC)nn2)=O)CC(F)(F)CC1CNC(=O)CC1CC(O)C1(C)C c1(Cc2cnc(C(=O)NCCc3cn(CC4CC4)nn3)s2)ccc(Br)cc1 C1(NC(C(c2ccc(C)cc2)=O)=O)CN(C(=O)C(C2(O)CCCC2)F)CCC1C c1(-c2ccc(C3(C)ON=C(C(C)C)C3)cc2)ccnc2ccc(C(=O)C3CC3)cc12 C(=O)(C1=CCCCC1)N1CCC(CC)C1C(=O)NCc1nc(C)c(C)[nH]1 CC1(C)CCOC1CC(N1CCC(CNC(c2c(F)cnn2CCN)=O)C1)=O C(C(=O)NC1CCOC1)(C(C)C1CCC1)N(CCC#C)CC c1(OC)ccc(C(=O)NC(C2CC(NC(=O)CCn3cccn3)C2)C)cc1 O=C1CN(CC(N2C(C(=O)NCC3CSC3)CC3CC23)=O)CCN1 c1(C(=O)NC(C2CCN(C(c3cnc(NC(C)C)nc3)=O)C2)C)ccc(F)nc1 N1(C(C(CCCC)O)=O)CCCC12CCN(C(=O)CC1CC3CC1C3)CC2 C(CCCCC(=O)NCCC1=CCCC1)NCCCC(=O)OC.Nc1ccc(C)nc1 CC1CCC(C)(C(=O)NCC2(CNC(=O)CC3CC3)CC23CCC3)CC1 C(CC(O)C(F)(F)F)NC(CCNC(c1n[nH]c(=N)[nH]1)=O)=O N1(C(CC=CC(C)(C)C)=O)Cc2n[nH]cc2C1C(=O)NC(C(N)=O)C1CCCC1 N(C1CCc2ccc3c(c21)CCO3)C(CCC1C(C)C1)C(=O)NCC1CCOC1 N1(C(=O)Nc2c(OCC)noc2C)CCCc2ccc(NS(C)(=O)=O)cc21 N1(C(CC2(C)CCOCC2)=O)CCC(C2CC2)C1C(=O)NC12CCCN(CC1)C2 C1(CNC(c2nc(Br)cs2)=O)CCCCN1C(c1ccc(C(F)(F)F)[nH]1)=O c1(NCC2(COC)CCCOC2)ccc2ccc(Cl)c(C)c2n1 C(=O)(C(O)C(C)(C)C)N(C1CN(C(c2cnc(C3CCCCC3)nc2)=O)C1)C N1(C(C23CC(CN(C(C4CCCOC4)=O)C2)C3)=O)CCC12CCCSC2 C1(CC(=O)NCC=CCNC(C(c2ccccc2)N(C)C)=O)CCC(=O)N1 C=C=CCCC(=O)NCC1CC(NC(c2cccc(-c3ccoc3)c2)=O)C1(C)C C(=O)(C1=C(Cl)CCCC1)NC(C)C(C)C(N1CCC(C2CC2)C1)=O N12CC(C)(CC1(C)C)COc1cc(sn1)Cc1cc(ccn1)C2=O.CO C=CCC(C)(CC=C)NC(=O)CC(C1CC1)NC(c1nc(C)ccc1C)=O C12(CNC(CC(COC)C)=O)CCCC1N(C(C13CC(F)(C1)C3)=O)CC2 C(=O)(CCCC(=O)N1CCCC1CNC(C1CCC(N=[N+]=[N-])C1)=O)OC Cc1c(C(=O)NCC(C)NC(=O)C(O)Cn2cncn2)ccn1C(C)C Cc1ccc(C(C)(C)CC(=O)N2CCC(NC(=O)C(C(C)O)N(C)C)C2C)cc1 c1(CN2CCC(CNC(c3c(Cl)cccc3Cl)=O)C2)cc(F)cc(F)c1O c1(C(=O)NC2(N(C(=O)OC(C)(C)C)CC)CC2)ccc(C)c(I)c1 c1(NC2C(C)CN(C(=O)Cc3csnn3)C2)ccccc1[N+](=O)[O-] C(CCO)(C(C)(C)O)NC(c1cc(CNC(c2c(C)snc2)=O)ncc1)=O N1(C(CNC(N)=O)=O)CCN(C(=O)CN(C(=O)C=Cc2cccnc2)C2CC2)CC1 n1(CC)ccc(C(=O)NC(C)(C)C(C)NC(c2cnsc2C)=O)cc1=O C1(NC(c2n(C)cc(F)c2)=O)CN(C(=O)Cc2ccccc2O)CCC1(F)F C#CCC(C)(C)C(=O)N1CCC(CCCNC(c2cccc(C(C)=O)c2)=O)CC1 c1(C(N2CCOCC(NC(c3n(C)cc(Cl)c3)=O)C2)=O)nc2c(s1)COCC2 N1(C(C2CCC2)=O)CCCC2CCN(C(C3(N4CCOCC4)CCC3)=O)CC12 CC1CCC(C)CN1S(=O)(=O)CC(C#N)C1CCOCC1 CCCC(O)CC(=O)NCC1CC(F)(CNC(C2(CF)CC2)=O)C1 CCC1=NOC(C(=O)NCC2(NC(=O)Cn3cc(-c4ccc(Cl)cc4)nn3)CC2)C1 C1(C#CC(=O)NC2CCCC(CNC(=O)CCc3cc(C)no3)C2)(CC)CC1 c1(-c2n(CC)ncn2)ccc(C(N2CC(NC(C3CC3C)=O)C(C)C2)=O)cc1 Cc1c(CC(=O)N(C)Cc2cn(-c3ccnc(F)c3)nn2)cccc1[N+](=O)[O-] c1(C(N2C(C(C)C)C(NC(=O)C(O)CC3CC3)CC2)=O)csc2cncn12 c1(C(=O)NC2C(NC(=O)C=C3CCSCC3)COCC2)cccc2c1NCCC2 N1(C(CS(CC)=O)=O)C2CCC1C(C(=O)NCC1C3CCCOC13)C2 Cn1cc(C#CCNCc2c(-c3ccccc3)cnn2C)cn1 CC(CCCc1ccccc1)C(=O)NCCCOCCNC(=O)CCCN(C)C c1(C(=O)NC2CN(C(c3cnc(C)[nH]3)=O)C2)ccc(Br)c(C)c1F C(c1ccc2ccccc2n1)=CC(=O)NC1CCC(CNC(CCCC#N)=O)C1 C1(NC(CC=C)=O)(CO)CCN(C(c2cccn2CCC#N)=O)CC1 C1(NC(=O)C=CCN2CCCC2)COC2(CCN(C(=O)CCF)CC2)C1 C(C)(c1ccncc1)=CC(=O)N(C)CC1OCCN(C(CC)=O)C1 C(=O)(CCCF)N(C1CCN(C(=O)CSc2n[nH]c(C)n2)C1)CCC C1(C(N(CCCCN(C(C(CC)OC2CCCC2)=O)C)C)=O)CC(F)C(=O)N1 CN1CC(NC(C2CC(C)(NC(=O)CCc3cn(C)nn3)C2)=O)C2(CC2)C1=O c1(C(N2CC=CC(NC(C3ON=C(CC)C3)=O)C2)=O)cn(C)c2ccc(Cl)cc12 N1(C(C=CCCC)=O)CCC2(CC2)CC1C(=O)Nc1cc(C#N)ccc1O CC1=CCN(C(=O)C=Cc2ccccc2)CC1.C1(C(=O)O)(N)CC(CO)C1 CCC(CC(C)C)C(=O)NC1CC12CC(NC(=O)Cc1nn(C)cc1Cl)C2 CC1(NC(C2CC2(Cl)Cl)=O)CC(NC(c2ccc(-c3ccccn3)s2)=O)C1 Cc1cc(C)c(C(=O)NCCSCC(=O)N(CC(C)(C)C)C(C)C)s1 CC(CNC(=O)CC12CCCC1C2)(CO)NC(=O)CSc1nnc(S)s1 C(CC)(C(=O)N1CC=CC1C(=O)NC(C)C(=O)NC(C)C)OCC C1(CCOC)CN(C(c2ccc(Cl)[nH]2)=O)CCN1C(C1CCCC1C)=O C1(C(=O)NC(C)(C)C)CN(Cc2ccccc2SC(C)C)CC2C=NN=C12 CCC(CC(F)(F)F)C(=O)N1CC(NC(=O)C=C2CCC2)C(C(F)F)C1 Cc1cc(C(=O)NC2CCC(NC(=O)Cc3c(C)noc3Cl)CC2)nc(O)n1 C1(CC)CC(NC(=O)NCCC2(CC3CCC3)CC2)C1 C1(NC(C(F)=CC)=O)CC(c2ccccc2)(NC(c2cnc(OC)s2)=O)C1 c1(C(=O)NCC2N(C(c3c(Cl)cnc(SC)n3)=O)CCC2)cccc2[nH]ccc12 C1(NC(c2c(C)nncc2)=O)CC2CC(C1)N(C(=O)CN(C)C(N)=O)C2 C1(COC(C(CC)CC)C)CC12CCN(C(=O)OC(C)(C)C)CC2 C1(C(N(CC(C)(C)C)CCC)=O)CCN(C(=O)CCc2cnc(C)o2)O1 Cc1ccc(NC(C2(C)CCN(C(C3CCCN3C)=O)C2)=O)c(O)n1 C1(C(=O)NCC2CC(C)(C)CN2C(=O)CC(F)(F)F)CC2CCCCCCC12 N1(C(=O)CN2CCCCC2)CCC(C2CCCN2C(C2CCCOCC2)=O)CC1 C(C(C(F)(F)F)n1cccn1)NC(N1CCCCC1c1ccc(F)cc1)=O C1(CC)CNC(=O)CN1C(=O)CN(C1CC(C#N)C1)C(C1CC1CC(C)(C)C)=O Cc1ccc(-c2nc(CCOc3ccc(Cl)cc3)nn2CC2CC2C)nn1 c1(COC)ccoc1C(=O)NC1COCC1C(=O)NC1CCC1(C)C CC(C)CC(C)(CNC(=O)CC1CCN(C)C1)NC(C1CC(C)(F)C1)=O c1(OC)ccc(C)cc1C=CC(=O)NCC1N(C(=O)COC)CCCC1(C)C CC(O)(CNC(C1CCCCN1C(=O)CCn1cnnn1)=O)CC(=O)O N1(C(=O)NC2CCC(F)(F)CC2O)CCC(F)(F)C2(CCOC2)C1 O=S(=O)(c1ccc(NC2CCN(CCF)C2)c(Cl)c1)NCC12COC(CF)(C1)C2 C(=O)(CC(O)CN(C)C)NCC(CC)NC(=O)C(c1ccc(OC)cc1)(C)C C(=O)(C(Cc1ccccc1)CC)N(CCCNC(COC(CC)(C)C)=O)CCO CC(CS(C)=O)C(=O)N1CCC(=CCNC(=O)Nc2nn(C)cc2Br)CC1 c1(C(=O)NC(C)CCNC(=O)CN(C)C2CC2)cc2c(nc1O)C(C)(C)CCC2 C1(c2ccc(C)nc2Cl)CC2(C1)NC(=O)N(CCC1CCCCO1)C2=O C(CN=c1nc(N2C3CCC2CN(C)C(=O)C3)c2c([nH]1)CSC2)(C(C)C)OC C(CC)(CC(=O)NC1CC1O)NC(C(CC)=CC)=O c1(CCNC(C2C(CNC(C=C(C)C(C)C)=O)CCC2)=O)cc(C)n(C)n1 C1(CNC(C=C(C)C(F)F)=O)(CNC(C2(C#N)CCCO2)=O)CCOCC1 c1(C(N2CCC(CNC(=O)C(F)(F)c3nccs3)C2)=O)nccc2occc12 CC1CC(C(=O)NCC2(CCNC(=O)CC3C(C)(C)C3(C)C)CC2)CC(C)(C)C1 c1(OC)ccc([N+](=O)[O-])c(NC2CC(C)N(C(=O)C(c3ccccc3)OC)C2)n1 C(=O)(C(C(C)(C)O)NC(c1n[nH]c(C)c1Cl)=O)NCCCCC#C c1(C(=O)Nc2ccc(NC(CC(CC)C)=O)nc2)ccc(C)cc1OC c1(CC)nc(C)oc1C(=O)NCC(C1CC1)NC(=O)C=CC1CCCC1 c1(C(C)NC(C(=O)OC)(C)Cc2ccccn2)cccc(Cl)c1C Cc1nc2c(s1)CC(C(=O)NC(C)(C)CNC(=O)COC(C)(C)C)CC2 C1(CNC(CSCC=C)=O)(NC(=O)C(C)N(C)C(=O)NCC)CCC1 C(=O)(C1=CC(O)C(NC(C23CCC(CC2)C3)=O)C1)NCC1(C)CC1(F)F C1(CCCC)CN(C(=O)CSCC(=O)Nc2ncc[nH]2)CCN1C(=O)CC(F)F Cc1ccc2c(C(=O)NC(C)(C)CNC(c3nnn(C)c3N)=O)ccnc2c1 C12(C(=O)N(C3(C)CCC(C)C3C)CC)COC(=O)N1CCN(C(=O)OC(C)(C)C)C2 CC1C(C)N(C(c2ncccc2F)=O)CCN1C(=O)CCCC(F)(F)F CC(C)C(CN(C)C)C(=O)NCC(C)N(C)C(c1ccccc1N1CCCC1)=O CC1CCCN(C(=O)COc2ccc(F)cc2Cl)C1CNC(=O)CC1CCC1 c1(OC)cc(F)ccc1C(N1CCC(O)(CC#N)C1)C(=O)NC(C)(C)C N1(C(C=Cc2cc(C)no2)=O)CCCC(C(=O)N(CCCO)CCCO)CC1 O=C1CCC(C(=O)NCc2ncccc2C(=O)NCCOCCCF)CC1 C1(C(N2CCC(CN(C)C(c3cccnc3)=O)C2)=O)CCn2c(cnc2Br)C1 O=S(=O)(c1ccc(NC2CCCC2O)c(Cl)c1)N1CCN(c2ccccn2)CC1 C1(CNC(COC)=O)CCN(C(=O)COc2cnn(C)c2)CCC1(F)F N1(C(C(C)(C)CO)=O)CCC2(CCC2NC(C23C4CCC(CC24)C3(F)F)=O)CC1 C1(NC(C(CCC)N(C)C)=O)CC2(CCN(C(=O)COCc3cccnc3)C2)C1 C(=O)(CCCS(C)(=O)=O)NCC1(CNC(c2n(C)c(S)nc2)=O)CCCC1 c1(C(N(CCNC(=O)C=CC(C)(C)C)CC)=O)cnn2c1OCC(F)C2 c1(CC)nc(C(=O)N(C2(C(N3CC(O)(c4nn[nH]n4)C3)=O)CC2)C)co1 N1(C(c2cc(Br)no2)C(=O)NCC(=C)C)CCCCc2cc(OC)ccc21 C1(CN(CCNS(CC)(=O)=O)C)CCCCN1C(=O)Nc1ccsc1 c1(C(=O)NCCOC2CN(C(c3cccc(OCC)c3)=O)C2)ncn2c1CCC2 NS(=O)(=O)C1COCCN(c2ccnc3c2CCCC3O)C1 C1(CC(=O)NC(C)(C)CNC(c2[nH]ccc2-c2ccccc2)=O)CC2C=CC1C2 c1(OCCCC)ccc(CCN(C(C2CC(n3ccnn3)C2)=O)CC)cc1 c1(C(N2CCN(C(CCCC#CC)=O)C(CCO)C2)=O)sc(S(N)(=O)=O)cc1C C1(OC(C)(C)C)CC(CC(N2CC(=CC(=O)Nc3ncc(Cl)s3)C2)=O)C1(C)C C1(C(=O)NC2CC(CNC(C3CC(OC)C3)=O)C23CCC3)CC2(COC(=O)N2)C1 C(CC(C)(C)C(=O)NC1CCC(CCNC(=O)C(C)C(C)(F)F)C1)OC N1(C(C(CCC)O)=O)C2CCC1CN(C(C1(c3cncnc3)CCOCC1)=O)C2 C12(CNC(N3CCN(CCC=C)CC3)=O)CC(CO)(CCO1)C2 C(=O)(C(CNC(C1CCC(OC)C1)=O)CC1CCCC1)NC(CC)(C)COC N1(C(C(C=C)O)=O)CCCCC1CCC(=O)NCCCOC(=O)NC c1(C(=O)NCC(CC)NC(c2cccc(SC)n2)=O)ccc(-c2cnco2)cc1 N1(C(C(CC)N(C)C)=O)CCOC2CCN(C(=O)C=C(C)c3cnn(C)c3)CC12 S(=O)(=O)(c1csc(C(N2CCCC(NC(c3cnc(N)c(Cl)c3)=O)C2)=O)c1)NC CN1CCN(C)CC(C(=O)NC2CC3(CCN(C(=O)C(O)CC(F)(F)F)C3)C2)C1 C1(OC)CN(C(=O)OC(C)(C)C)CCC1NC(=O)C(c1ccc(Br)c(F)c1)C C(=O)(C(C)(C)NC(=O)C(C1CC1(Br)Br)N(C(C)C(=O)OC)C)NCCC N1(C(C(CC(C)C)O)=O)CC2(CNC(=O)Cc3cncnc3O)CC1CCO2 C1(CC(=O)NC2CC(CC)C2)CCN(C(=O)C(C)S(N)(=O)=O)C1(C)C Cc1cc(Cl)ncc1NC(=O)NC1CN(C(C)(C)C)CC1c1ccc(F)c(F)c1 CC1COC(CO)CN1C(=O)CC1CCN(C(=O)Cc2cncnc2O)CC1 c1(C(=O)NCC2C(NC(C3(CC)CCCCC3)=O)CCC2)ccc(O)c(O)c1 c1(CNC(C2CCCC(NC(CN(CCOC)C)=O)C2)=O)ccc(F)c(F)c1 c1(OCC)cc(Cl)ccc1NC(N1CCNCCC1C)=O CC1CN(C(=O)C(c2cc(Cl)ccc2Cl)(F)F)CCC1N1CCCC1 c1(C(=O)OC)ccnc(N2CCN(C(=O)CC3OCCC3C)CC2)c1[N+](=O)[O-] CCCCC(C)C(=O)N1CC2(CO)CC1(C(=O)NC(CC(=O)NC)C1CC1)C2 C1(CC)(NC(=O)C=Cc2nc(C)c(C)[nH]2)CCN(C(=O)CS(=O)(=O)NC)CC1 C(C(=O)NCc1ncc(C)[nH]1)(C(C)CC)N(C(CCC=C=C)=O)C N1(C(CC=C)=O)CCC(C2(O)CN(C(=O)CCc3ccnc(C)n3)C2)CC1 CC(CC(=O)NCCCCCCNC(C1CCN(c2nc(=N)[nH][nH]2)C1)=O)C(F)F c1(C(=O)NCC2CCC(NC(CCNC(C)=O)=O)C2)ccc(Cl)c(N)c1 CCCCCCC(CC)C(=O)N1CCN(c2ncnc3[nH]ccc23)CC(O)C1 C1(C)(NC(c2c(OC)c[nH]n2)=O)CCN(C(=O)C(C)n2ccnc2)CC1 c1(C(=O)NC(CNC(C2CC(CC)(CC)C2)=O)C)cc(O)ccc1N c1(C(=O)NCC23CCC2CN(C(C2CC2F)=O)C3)c([N+](=O)[O-])cnn1CC(F)F CC(C)C#CC(=O)NC(C1CCCN1C(=O)C=Cc1ccccn1)C C(CCCC(C)(C)C(=O)NNC(=O)C(O)C1CC1)NC(CNC(CC)=O)=O C1(CC)C(C(=O)NCC2CC(=O)N(C)C2)CCCN1C(c1ncccn1)=O N1(C(c2c(CCC)n[nH]c2)=O)CCC2CC2(C(=O)NC2CCN(C)C(=O)C2)CC1 CON(CCC(=O)N1CC2CCCC2(NC(=O)C(C)CF)C1)C(=O)OC(C)(C)C C1(C(N2CC(CCNC(c3ccc(C(N)=O)[nH]3)=O)(OC)C2)=O)C2CCCCC12 Cc1c(C(=O)NC2CC(CO)N(C(=O)CCC3CCCN3C)C2)cnn1CCO CC(CN(C)C)CC(=O)N1CC(O)(CCNC(=O)CC2CC(F)C2)C1 C1(CC)CCCN(C(=O)CCC(C)N(C)C)C1C(=O)NC1CC(CO)C2CC12 N1(CC)CC(C)(C)OC(=O)C1CC(=O)NCC(CC(C)C)NC(C1CC(O)C1)=O C(=O)(C(C)(C)C(=O)N(C)C)NCC(C)CNC(c1cncn1C1CC1)=O CC1CC2CCC(C1)N2C(C1C(C)CN1C(=O)C(C1CCOCC1)=O)=O CC(C)C(N=[N+]=[N-])C(=O)NCC1CC(C(=O)N2CCC(OCCO)C2)=NO1 N1(C(C2(CNC(C3CC(CC)C3)=O)CC3(CC3)C2)=O)CC(C)OC2(CCC2)C1 C(C)(C)(CC(F)C(=O)NCc1ccc(CO)o1)NC(CC1ON=C(C)C1)=O C(=O)(C(F)C(C)CNC(=O)Cc1csnn1)NCC(=O)NCC#C c1(C(=O)NC(C2CCN(C(C(CC=C)C)=O)C2)(C)C)noc2ncccc12 C#Cc1cccc(C(=O)NC2CCC(NC(=O)CCc3ccncc3)CC2)c1F Cc1cc(C(=O)NCC=CCNC(=O)C(C)(C)c2ccn(C)n2)cnc1C c1(C(=O)NC(CNC(c2cn(CCC)nn2)=O)C2CC2)cn(C2CCC2)nc1C c1(C(=O)NCC2(F)CC(CNC(CN3CC(C)C3)=O)C2)cc(F)c(F)c(F)c1F c1(C(=O)NC2(C)CCN(C(=O)CC3CCCCO3)C2)nnc2n1CCCC2 c1(CC)cc(C2CCN(C(=O)N(c3cccc(Br)c3)C)C2)ccc1C(F)(F)F c1(C(=O)NC(CC#C)C(=O)NC2CC(C#N)C2)ccnc(C)c1C C1(CNC(C(C(C)C)SC)=O)CN(C(=O)C(C2CCC2)C2CCC2)CC1(F)CO c1(C(N2CC(CNC(c3ccc(C(C)=O)o3)=O)C2)=O)cn(C)ccc1=O N1(C(c2ccc(COC)o2)=O)CCN(C(=O)C(n2nc(C)cc2C)C)C(C)C1 CC1(C)COCC(CC(=O)NCCOCCNC(C2CN(C(N)=O)C2)=O)O1 c1(C(C(=O)NC2CC2)N(CC(C)SC)C)csc(Cl)c1 C(=O)(CC(C)CF)NCC(C)CN(C(=O)CCc1ccc(Cl)cc1)C N1(C(C2(OC)CC2)=O)CCC(CNC(c2ncccc2CSC)=O)C(F)(F)C1 CC1C(=O)NCCN1C(=O)NC1CCC(C)C1 N1(C(CNC(c2coc(OC(C)=O)n2)=O)=O)CCCC(C)C1SCCOC C1(C(=O)OC(C)(C)C)(NC(C2(c3cc(O)n[nH]3)CC2)=O)CC(F)(F)C1 N1(C(c2cn(CC)nn2)=O)CCCC(C)(C)C1C(N1CCC(C(N)=O)CC1)=O CON(CCC(=O)NC1CC2CC3C(C2)C13)C(=O)C1(C)CCCCCC1 C1(NC(C2=C(C)OCC2)=O)COC2(CCN(C(C3C=CCC=C3C)=O)C2)C1 c1(OCCC(=O)NC2CCCC(CNC(CC(C)(F)F)=O)C2)ccc(F)c(F)c1 N1(C(C(C=C)(C)C)=O)CCC2(CCCN(C(c3nnc4ccccn34)=O)C2)CC1 C1(CNC(C(C(=C)C)(C)C)=O)COC(C)(C)CN1C(=O)C(CC(C)C)C1CCC1 c1(C(=O)NC2C(NC(c3cc(C)n(C(F)F)n3)=O)C2)nccc2ccccc12 N1(C(c2c(C)ncs2)=O)CC2CCCC(C1)C2C(=O)NCCOC(C)C C1(C(N(CC)CC2CCN(C(C3CC3C)=O)CC2)=O)Cc2ccccc2S1 C1(CN(C(=O)Cc2cnc[nH]2)C)CN(C(=O)Cc2cccc(O)c2)CC12CC2 C1(CNC(c2ncc(NC(C(=O)N(C)C)=O)n2C)=O)CCC2(CCC2)CC1 Cc1ccc(C(=O)NC2(CO)CCCN(C(C3(C)CC3C(F)(F)F)=O)C2)c(O)c1 c1(OCC=C)cccnc1NC(c1csc(C(F)F)c1)c1nnnn1C(C)(C)C n1(COC)nccc1C(=O)NC1COCC1CNC(=O)CC(C)=C(C)C C12(CNC(=O)Cn3nccn3)CCC(CC1)N(C(c1ccc3nc[nH]c3c1)=O)C2 C(CCC)(C(=O)N1CC=CC1CNC(c1cc(C(F)F)ncn1)=O)=CCC N1(C(C2ON=C(C)C2)=O)CCC=CC1C(=O)NCc1cccn1C N12CCN(CC1)C(C)CNC2=O.c1(NC(c2sccc2C(N)=O)=O)ccccn1 c1(OC)c(C)cc(C(=O)NC2CCN(C(=O)COCC3CC3)C2C(C)C)cc1Cl C1(NC(C2CC3(CCC3)C2)=O)CCCC12CCN(C(C1(O)CCCC1)=O)C2 C1(NC(C2CN3CCC2CC3)=O)CCSC12CN(C(=O)C(F)C1CCOC1)C2 c1(OC)cc(C)ccc1C(N1CCC(C)(NC(C2CCCSC2C)=O)CC1)=O S(=O)(=O)(c1ccc(Br)cc1)NCCNC(C(C)CC(C)(C)C)=O Cc1sc(O)nc1C(=O)NC(C(C)NC(c1ncccc1F)=O)C(C)C C1(C)(CSC)CCN1C(=O)NC1CCC(N(C)C(=O)OC(C)(C)C)C1 C1(N(C(c2cccnn2)=O)CC)CCCN(C(c2nc(C)c(Br)s2)=O)CC1 C(C1Cc2ccccc21)NC(C(C1CCC1)NC(c1ccnn1CCF)=O)=O c1(CC)ccc(OC)cc1C(N1CCN(C(=O)Cc2nccn2C)CC1CF)=O C(=O)(C1=CCCOCC1)NC(C1CCCC1)CNC(c1c(C)nn(C)c1C)=O N1(C(C2CC(C)C2)=O)CC=CC1(C)C(N1CCC1CC1CCCC1)=O C#CCC(C)C(=O)NC(C)CC(C)NC(C12CC(C1)C(C(F)(F)F)O2)=O c1(C(N2CCN(C(c3cnc(CC)s3)=O)CC2CC)=O)cc(Cl)c(N)c(Cl)c1 c1(C(=O)NCCC(C)N(C(=O)CC2CCCC2)C)ccc2cc[nH]c2c1 C1(C(N2CC(C(C(=O)NCCCC3N(C(C)=O)CCC3)O)C2)=O)CCC2(CC1)CC2 c1(C(C)C(N2CCC(N(C(=O)C(=O)NC(C)C)C)C2)=O)ccc(Br)cc1F CC1CN(C(=O)Cc2cccc(Cl)c2)CCC1N(C(=O)CCn1ccnc1)C Cc1cc(C(=O)NCC2CC(O)CN2C(c2cnn(C)c2)=O)nn1C(F)F C(=O)(CC1CNc2ccccc21)N1C(CNC(C2CCC3(CC2)CC3)=O)CCC1 CC1CN(c2ccccc2NCc2cccn2C2CCCC2)CC(C)O1 c1(OC)ccc(NC(=O)CC(O)CNC(=O)C(C2CCCC2)OC)c(C)c1 N1(C(C2C(CCC)CCC2)=O)CCSCC1CCNC(c1ccn(C(F)F)n1)=O N1(C(C2ON=C(C)C2)=O)CC2CC1C2CNC(c1ncccc1F)=O c1(C(N2CCCC(CNC(c3onc(C)n3)=O)CC2)=O)sc2ncccc2c1N CC1C(NC(=O)CCc2ccn(C)c2)CCCN1C(c1nccc(Cl)c1F)=O C12(C(N3CC(C#C)(N(C)C)C3)=O)CC(CCO1)N(C(c1cc3ccccn3c1)=O)C2 c1(C(=O)NCCCNC(C2C(OC)CCC2)=O)cccnc1O C1(CC)CCOCCN1C(=O)C(CC1CC1)NC(=O)CC1(C)OCCO1 C1(C(C(N)=O)NC(C2CC2Cl)=O)CCC(F)(F)CC1 Cc1nccc(C(N2CCOCC2CNC(=O)C(F)(F)c2ncccn2)=O)c1C C1(OC(C)C)CCN(C(C2CN(C(C3CC3(F)Cl)=O)CC2C(C)C)=O)CC1 N1(C(C(C)OCCOCC)=O)CCCC(C)(CNC(=O)CCCN2CCCC2)C1 c1(CC(=O)N(C2CCN(C(c3cccc(CS(C)=O)c3)=O)C2)C)cn(C)nc1Cl N1(C(c2nc(CCCCC)sc2)=O)CCN(C(=O)CC2COCCO2)C(CO)C1 CC1C(NC(=O)C(F)(F)F)CCCN1C(=O)C(N1CCCCCC1N)=O C1(CNC(C2(CC)CNC(=O)C2)=O)CC(C)CN(C(C2CC2C(N)=O)=O)C1 C1(C(=O)NCCC2(CNC(c3ccc(CSC)cc3)=O)CC2)CCC2(CCC2)O1 C(=O)(CCCS(C)(=O)=O)NC(C1N(C(c2n(CCC)ncc2Cl)=O)CCC1)C C1(NC(c2c(C)nccn2)=O)CN(C(=O)Cc2cnoc2)Cc2ccnn2C1 O=C(CCCCCBr)N1CCN(C(C2(c3ccc(Cl)cc3)CC2)=O)C(CO)C1 c1(C(=O)NC(CN(C(Cc2cc(OC)no2)=O)C)C)[nH]cc2c1CCS2(=O)=O C(=O)(C(C)C(C)(C)C)NCC1C(NC(C(=O)Nc2ccc(OC)cc2)=O)CC1 C12(CNC(CC3(OCC)CC3)=O)CCCC1CN(C(c1ncnn1CC)=O)C2 CC(N=c1[nH]c2c(c(=NC3COC4(CCCC4)C3)[nH]1)COC2)c1ccc[nH]1 N1(CCCN(C)C(C2(C)CC3CC3C2)=O)CCN(C(=O)NC)CC1.C(C)(C)(C)O N1(C(C)Cc2ccccc2Cl)CCC2(CC1)CC2C(=O)NC(C)CCO Cc1n[nH]c(C)c1CC(C)C(=O)N(CCNC(C1(O)CC(C)(C)C1)=O)C1CC1 CC(C)(C)C(CNC(c1cc(C#N)ccc1N)=O)C(=O)N1CCC(O)C(O)C1 C(C(=O)NC(C1(O)CN(C(=O)CC(C)(C)C#N)C1)C)(C(C)(C)C)SC Cc1ccc(OCCC(=O)NCC2CCCN2C(=O)CC2CCN(C)C2)c(C)c1 n1(CC)nc(C)c(CC(=O)NCC(O)CN(C)C(c2ccn(C3CC3)n2)=O)c1C N1(C(c2c(-c3cn(CC4CC4)nn3)cc[nH]2)=O)CCC(n2cc(I)cn2)CC1 C1(NC(C2N(C(C(CC=C)CC)=O)CCC(=C)C2)=O)CCC2CC1C2(C)C c1(OC)ccc(C(=O)NC2COCC2NC(C2(CF)CC2)=O)c(F)c1Cl C1(N(C(c2csc(CNC(=O)CCCF)c2)=O)CC)CCCCC1C C(CO)(CC(C)(C)C)NC(C(CNC(COC)=O)CC1CC1)=O N1(C(C(C)(C)NC(CCCOCC)=O)=O)CC2(CCC2NC(c2cnn[nH]2)=O)C1 N1(C(C2C(C)C2C)=O)CC(NC(=O)COCc2ccncc2)CC(O)C1 C(CN=c1[nH]c(=NCC23CCCCC2C3)[nH]c2c1COC2)Sc1cncc(Cl)c1 C(=O)(C1=C2CCCN=C2NN1)N1CC(NC(c2cc(C)nc(C)c2)=O)C(C)(C)C1 c1(N2CCC(CC)C2)nc(=NC2CN(C(C3CCC3)=O)C2)[nH]c2c1cnn2C C1(C(=O)OC)=NC=CC(c2ccccn2)=NN1C(C1CCC(OC(F)F)CC1)=O c1(C(N(CCNC(=O)C=CC(N2CCOCC2)=O)CC)=O)cnnc(C)c1 Cc1cc(C(N2CCC(C)(CNC(=O)C(C)C(C)(F)F)CC2)=O)c(C)cn1 C(=O)(C(C)(C)CCC)N1CCC(O)(CNC(CCN(CCC)C)=O)C1 N1(Cc2c(OC)cccc2)CCC2CN(C(=O)Nc3cccc(F)c3O)CCC12 C12(NC(=O)C3=CCC3)CCCC1N(C(=O)CCc1cccc(F)c1F)CCC2 c1(OC)cc(C(=O)NC2CC(CNC(C3(O)CCCCC3)=O)C2(C)C)cc(F)c1 c1(OC)cnccc1C(=O)NC1CC1NC(c1nc(C)oc1C)=O c1(C(=O)NC2CN(C(C(C)OCC=C)=O)CC2CC)c(CC)cccc1C C1(CNC(c2c(OC)cc(SC)cc2)=O)CC2(CCC2)CN1C(=O)CCC1CC1 c1(C(N2CC3CC2CN3C(C2CCCC2)=O)=O)cnc(C(F)(F)F)c(F)c1 N1(C(c2[nH]cc(C(C)(C)C)c2)=O)CCCC(CO)(NC(c2ccn(C(F)F)n2)=O)C1 C1(F)(C(N2CCC(CNC(c3c(C(C)C)nn(C)c3)=O)C2)=O)CC12CCCCC2 N1(C(C(c2c(C)cncc2)C)=O)CCC2(CC1)CCN(C(C1CN(C(N)=O)C1)=O)C2 c1(NC(C2CC(NC(c3c(C)n[nH]c3C)=O)C2)=O)c(F)c(F)nc(F)c1F CCC(CC(=O)NCC1CCC(CNC(C2CS(=O)(=O)C2)=O)CC1)CC(F)(F)F c1(SC)ccc(C(=O)NCCC(C)NC(=O)Cn2ncccc2=O)cc1 N1(C(c2cc(C)nc(C)n2)=O)CC(C)(C)OCC1CNC(c1cc(C)on1)=O C1(C(N2CCC(CN=[N+]=[N-])C2)=O)CN(C(=O)C(F)C2CCCC2)C2(CCC2)C1 CC1(CNC(=O)CCCC2CCCC2)CCN(C(=O)CCC2NC(=O)NC2=O)C1 CCCC(C(=O)NC(C)(COCC)CO)NC(c1ccc(OCC)nc1)=O N1(C(c2cncc(C(N(C)C)=O)c2)=O)CCC(C)(C)C1CNC(=O)NC1CC1Cl Cc1ccc2c(C(=O)NC(C3CCCN3C(C3CC3CF)=O)C)c[nH]c2c1 CCC(CC(F)(F)F)C(=O)NC1(CCOC)CCN(C(c2sccc2CO)=O)C1 N1(C(CC)=O)CCC(F)(CNC(=O)C2=CCCOC2)CC1 c1(C(N2CCC(CCNC(C3N=C(C)SC3)=O)CC2)=O)ccnc2ccsc12 C1(NC(=O)CC2CC3(CCC3)C2)CC2CCC(C1)N2C(=O)Cc1ccco1 C(C(C)(C)CO)(c1ccccc1)NC(=O)NC(c1ccc(C)o1)CC Cc1cc([N+](=O)[O-])ccc1C(=O)NCC(C)NC(=O)C(C)(C)CO CC1CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)C(C)CN1C(=O)CC(C)(C)N(C)C Cc1nc(O)[nH]c1C(=O)NCC12CC(NC(C3C4CCC(F)C34)=O)(CO1)C2 C(=O)(CCCCCCNC(=O)CC1(C#N)CC1)N1C(CC)(CO)CCC1 c1(-c2cn(C)nc2)cncc(C(N2CCC(N(C(=O)CS(C)(=O)=O)CCO)C2)=O)n1 c1(C(N(CCNC(C2(C)CC2F)=O)CC2CC2)=O)cnc(S)n1-c1ccccc1 c1(C(N2CC(CNC(CCC3(C)CC3)=O)OCC2)=O)cc([N+](=O)[O-])sn1 CCCC(CC(=O)NCC(O)CC(C)C)NC(=O)C(O)CC1CCCC1 c1(C(C)(F)F)ccc(C(N2CC3CC3(NC(=O)C(O)Cc3cnc[nH]3)C2)=O)nc1 C#Cc1cccc(C(=O)NCC2CN(C(C3CC(F)C3)=O)CCN2C)c1F c1(C(=O)NC2(CNC(c3ccc(C)s3)=O)CC(OC)C2)c(C)noc1C N1(C(=O)C(F)C2CC2)CC(C2CCCN(C(c3ccc(=O)n(C4CC4)c3)=O)C2)C1 C#Cc1cccc(OCC(=O)N(CC(C)N(C(=O)C(O)C2CC2)C)C)c1 c1(CC2(C(=O)NCCN(C(=O)C(=Cc3cccs3)C)CC)CC2)ccc(F)cc1 Cc1ccc(N2CCCC(NC(=O)C(=O)NC3CCOC3C)C2)cc1 N1(C(CCN(C(c2cnc(CC)nc2)=O)CC2CC2)=O)CCCC(C2(C)CC2)C1 C1(C(=O)NCc2cc(C(=O)Nc3c(C(C)C)nn(C)c3)sc2)CC2C=CC1CC2 C1(CC=C)(NC(c2cnn(CCO)c2C)=O)CCN(C(c2ccc(C)n2C)=O)C1 C1(C(N(CC=CC(=O)NC2(C(C)C)CCC2)C)=O)CC(=O)OC1(C)C C1(C(=O)NCC(C)C(=O)NCCCn2cc(CO)nn2)(CC)CCCCO1 N1(C(C2CCN(C(c3c(NC)nccc3)=O)C23CC3)=O)C2CCC1CC(F)C2 N1(C(C(CNC(c2oc(C)c(CO)c2)=O)CC2CC2)=O)CC(F)(F)C(F)(F)C1 c1(C(=O)NC2CCC(CNC(C3(O)CCC3)=O)C2)ccnc(C(F)(F)F)n1 n1(CCSC2CC(C(C(=O)O)F)C2)cc(Br)cn1 C(=O)(CC(C)NC(N)=O)NC1C(C(=O)NC(c2nc[nH]n2)CC)CC1 N1(C(C=Cc2ccc(CC)o2)=O)C(C)C2CC1C2NC(=O)CNS(=O)(=O)NC N1(C(c2c(C)nc[nH]2)=O)CC2(CNC(c3cccc4oncc34)=O)CC(F)(C1)C2 c1(C(=O)NC2CCN(C(=O)C3=C(Cl)CCOC3)CC2)cc2c(F)cccc2s1 C(=O)(CCCCCC(C)C)NCc1cn(C2CC(NC(C)=O)CC2CO)nn1 C(N=c1[nH]c2cccnc2s1)C1C2CN(C(c3ccc(C#C)cc3)=O)CC21 c1(C(c2cccc(F)c2)NC(c2cnn(C)n2)CC)cccc(Br)c1 C1(C(N(CC=C)CC)=O)CCc2nc(C)nc(C(F)(F)F)c2C1 Cc1ncnc(O)c1CCC(N1CCCC(NC(C2(C#N)CC23CCC3)=O)C1)=O N1(C(C(C)Oc2ccc(F)cc2)=O)CCCOC(CNC(C23CSCC2C3)=O)C1 c1(C(=O)NC2C(CNC(C3=NOC(C)C3)=O)COC2)cccc2c1nc(O)n2C N1(C(C(CC)CC)=O)CCCOC(CCNC(=O)CN(C)S(N)(=O)=O)C1 c1(C(N2CC(CS(=O)(=O)C3CC3)C2)=O)cnn2c(F)cccc12 c1(C(=O)Nc2ccc(NC(C3CC3(F)F)=O)cc2F)cccc2cccnc12 c1(C(N2CC=CC(NC(C(C)OC)=O)C2)=O)cnc2c(c1)N(C)CCO2 c1(C(=O)NCCCNC(c2ccc(CC)o2)=O)ccc(N(C)CC)cc1 N1(C(C(c2cccc(Cl)c2)C)=O)CCC2C(CCCN2C(=O)CC2CSC2)C1 C(c1ccc(O)cc1)=CC(N1CC(C(C)NC(c2n[nH]cc2C2CCC2)=O)C1)=O C(CCNC(C1CCCCS1)=O)(C(=O)NOC1CCCC1)OC c1(CCC)n[nH]cc1C(N1CC(CC(F)C(=O)NCc2nccn2C)C1)=O C(N=c1cc(C)c(S(=O)(=O)NCCSCCO)c[nH]1)c1cc(C)c(Br)cc1 Cc1oc2ccccc2c1CNCC(N1CCC(O)C1c1ccccc1N(C)C)=O Cc1ccc2cc(C(=O)NCCC(N3CC(NC(=O)C(C)C)C(O)C3)=O)oc2c1 c1(C(=O)NCC2CN(C(C3(O)CC3)=O)CCO2)sc2ncccc2c1Cl C1(C2CCN(C(C3CCC(F)CC3)=O)CC2)(NC(c2cnn3c2CCC3)=O)CC1 CN1CCCC(C(N2CCC2(C)CCO)C(=O)Nc2ccccc2)C1 C(C)(c1cccc(Cl)c1)=CC(N1C(CCNC(COCCC)=O)CCCC1)=O Cc1nc(C(=O)NCC2(F)CN(C(C3CCC=CCC3)=O)C2)nn1C CC1CC(C(=O)NC23CC(C2)N(C(=O)CCc2ccncn2)C3)CCS1(=O)=O C12(C(=O)NC(C)CCN(C)C(c3nonc3N)=O)CCCC1C2(F)F c1(C(N(CC(C)NC(C(C)=CC2CC2)=O)C)=O)ccc(NC2(O)CCCC2)nc1 c1(CCC)nc(C)c(C(=O)NCC(C)(C2CCC2)NC(=O)C(C)C2CCCC2)s1 c1(C(=O)NC2CN(C(CCC(CCCC)C)=O)C2)cc2cccc([N+](=O)[O-])c2[nH]1 Cc1ccc(C(=O)N(CCNC(=O)C=CS(C)=O)Cc2ccc(Cl)nc2)nc1 C=CC(F)(F)C(=O)N(C)CC1CC(F)CN1C(=O)CC1(C)CCC1 c1(CNCC(C)NC(=O)CC2CCN2C(=O)OC(C)(C)C)ccc([N+](=O)[O-])nc1 CN1CCc2ccc(C(N3CC(C4CCOCC4)C3)=O)cc2C1 N1(C(CC)=O)CCC(C2(NC(c3ccc(-c4nnc(O)n4C)cc3)=O)CC2)CC1 N1(C(C(COC)(F)F)=O)CC2CCCC2(CNC(c2cc(C)nc(C)c2O)=O)C1 c1(C(=O)OC)cc(C(=O)NCCCNC(C2CC2Cl)=O)cc(C(C)C)c1 N1(C(Cc2nc(C)[nH]n2)=O)CC2(CCCC2C(=O)NCC2(CO)CCCC2)C1 Cc1ccc(CN2CC(CC(=O)O)CC2(C)C)c(Cl)c1.C1(C2C3C(C3)N2)CCC1 C(=O)(CC(C)(C)C)NC(C)C(c1ccccc1)NC(c1nc(C2CC2)cs1)=O CC(CC(=O)NCCc1ocnc1CNC(=O)CC1CCS(=O)(=O)C1)C(F)(F)F S(=O)(=O)(c1cc(C)cnc1N1CCC=C(Cl)C1)NC(CCC=C)CO c1(SC)cc(C(N2CC(N(C(=O)CCCNC(=O)C3CC3)C)C(F)C2)=O)oc1C CCC(C)C(C)C(=O)N1CCC(C)(NC(=O)CCCOC)C1 Cc1cncn1CC(=O)NCCN(C(=O)CNS(=O)(=O)Cc1ccccc1)C C#CC1(C(=O)NCC2(CCC=C)CCCC2)CCN(C(=O)OC(C)(C)C)C1 C1(NC(C2N(C(C)=O)CSC2)=O)CC(C)CN(C(=O)C(C)Cc2ccccc2)C1 c1(C(=O)OC)c(C)ccnc1NCC1(CCNC(c2ccc[nH]2)=O)CC1 c1(CC(N2CCC(CNC(=O)C3=CCCC3)C2)=O)ccc2nc[nH]c2c1 c1(C(=O)NCC(C(=O)NCCC(C2CC2)C2CC2)OC)cc(O)nn1C N1(CC)CCOC(C(=O)NC(C)(CNC(=O)COc2ccsc2)C(C)C)C1 N1(C(C2C(C(C)C)(CC)C2)=O)CCN(CC2CCC(=O)NC2)CC1 C(=O)(C(C(C)(C)C)NC(C1COCCN1C(c1cccc(SC)c1O)=O)=O)NC c1(C(N(C2CCCN(C(=O)C(CO)c3ccccc3)C2)CC)=O)ccn2c1CCCC2 S(=O)(=O)(c1cccs1)NCC(=O)NC1CCCC(CN(C(=O)CCCF)C)C1 N1(c2n(CCC=C)c(C3CCCCCC3C)nn2)CC(F)(F)CC1C S(=O)(=O)(c1ccc(C(C)(F)F)cc1)NCc1cccc(C(=O)NCCCCC)c1 N1(C(C(CC)F)=O)CC2OCCN(C(c3cnc(N)c(Cl)c3)=O)C2C1 Cc1c(C(=O)NC(C)CC(C)NC(c2cnns2)=O)c(C(F)(F)F)nn1C C1(NC(C(F)=CC)=O)CCCCN(C(C2CCCN(C(=O)NCC)C2)=O)CC1 N1(C(c2ccc(C)c(C)c2)=O)CCN(C(=O)Cn2cnc(Br)n2)C2CCC12 c1(C(=O)NCC2CC(OC)CN2C(C2(C)CCN(C)C2=O)=O)cccc(C)c1F N1(C(C=Cc2n(C)ncc2)=O)CCC2(NC(c3ccc(O)c(CO)c3)=O)CC2C1 C(=O)(CC(C)C(F)F)NC1CCC(N(C(CS(=O)(=O)NC)=O)C)CC1 c1(NC(COc2ccc(CC(N)=O)cc2)=O)ncc(C=NO)s1 C(=O)(C(F)(F)CC(C)C)N1CC(CNC(c2c(C)cccc2O)=O)C(C)CC1 CCCCC(C(=O)NC1(n2cnnn2)CC1)NC(=O)C1=C(Cl)CCC1 CC(O)C(C)(C)C(=O)NC(C)C(N1CC2CCCC2C1)=O C(=O)(C(F)(CNC(C1CCC2(CCC2)O1)=O)C(C)C)NC(C#CC)(C)C c1(OC(C)C)cccc(C=CC(=O)NCC2(NC(C3OCCO3)=O)CCC2)c1 c1(C(=O)NCCCN(CCO)C(C2CC23CC3(F)F)=O)cc(Cl)c([N+](=O)[O-])[nH]1 c1(C(N(CCC)CCNC(=O)C(C2CCCCC2)O)=O)nccc(N)c1Cl CC(C(C(=O)NC1COC1)N(C)Cc1nnn(C)n1)C1CCCC1 C1(NC(C(CCC)N(C)C)=O)COC2(CCN(C(C3(O)CCOCC3)=O)CC2)C1 C1(COC)(NC(C23CC(CC(F)F)(C2)C3)=O)CCN(C(C2(C)CNC(=O)C2)=O)C1 C1(CC(=O)NCC(CNC(c2ccc(NC)cc2)=O)OC)CCC(=O)NC1=O Cc1cnc(C(=O)NC2CCN(C(c3ccncc3N3CCCC3)=O)C2)c(F)c1 C1(C(=O)NCC(CN(C(=O)C=CCCc2ccccc2)C)O)COCCC1(F)F C1(C(=O)NC2C(O)CCN(C(C3C(OC)CCCC3)=O)C2)CN2CCN1C(C)C2 C(CCN=c1nc(N2CC=CCC2)c2c([nH]1)CCC2)c1cccc(C)c1 C1(CC)C(C(N2CCC(NC(C)=O)CC2)=O)CCN1C(=O)CC1CCCNC1=O c1(C(=O)NCCCN(C)C(c2ccc(C(F)F)nc2)=O)cc(Cl)nnc1O C1(CNC(CC=CCNC(CC2(CSC)CC2)=O)=O)CCCSC1 N1(C(CC(=O)NCC#C)=O)CCN(C)C(CNC(=O)C(CC)N2CCCC2=O)C1 N1(C(C(CC)SC)=O)CC(C(=O)Nc2cnc(O)c(F)c2)C2(CCC2)C1 C(CC(=O)N1CCCCC1CCCNC(c1nc(Cl)oc1C)=O)(C(C)C)OCC N1(C(C2CN(CCC)C(=O)C2)=O)CCCC(C2CN(C(=O)C(COC)OC)C2)C1 C1(NC(CC2(C=C)CCC2)=O)(CO)CCN(C(c2cnc(O)o2)=O)C1 CCCC(CNC(=O)C(C)SC)C(=O)Nc1ccc[n+]([O-])c1 Cn1ncc2cc(-c3cnc(C(=O)Nc4cc([N+](=O)[O-])ccn4)cn3)ccc12 C1(C(N2CCCC(N(C(C3(C=C)CC3)=O)CC)C2)=O)CC12CCSCC2 C1(CNC(CCC#C)=O)CCCC(NC(=O)C(N2CCC(O)CC2)C)C1 c1(OC)cc(C(=O)NC(C)(CNC(=O)CCCCC2CC2)C(C)C)cc(Cl)n1 c1(OCc2cn(C3CN(C(C4C(C)CCCC4)=O)C3)nn2)ccc(F)cc1[N+](=O)[O-] c1(C(=O)NCC2C3CN(C(CC(=O)OC)=O)CC32)ncn2ccccc12 C1(C(=O)NC(CN(C(CCSCCC)=O)C)CC)CCc2nn[nH]c2C1 N1(C(c2cncc(CC)c2)=O)C2CCC1CC(NC(=O)C(C1CCC1)OC)C2 C#CCCCCCC(=O)NCC1(F)CCN(C(=O)Cn2ncc(Br)c2C)C1 c1(C(=O)NC2(C)CN(C(C=Cc3ncn(C)c3)=O)C2)ccc2c(=O)cc[nH]c2c1 S(=O)(=O)(CC(=O)NCCC1(CNC(C2(C)CCCO2)=O)CCCCC1)NCC N(C1CN(C(C2CCC2)=O)Cc2ccccc21)C(C(C1CCCC1)OCC)=O N1(C(C(C)NC(N)=O)=O)C2CCC1C(C)C(NC(C1CCC3(CC1)CC3)=O)C2 CCCC(CC)CCC(=O)N(CC(C)(C)NC(c1nccc2occc12)=O)C CCCC(C(C)CC)N(C(=O)CC(O)(c1ccccc1)C1CC1)C C(=O)(C(CC(F)(F)F)NC(c1cc(F)ccc1OC)=O)N(CCCCCC)C N1(C(CSCCNC(C(C(CC)O)C)=O)=O)CCC2(CCOC2)CC1 c1(C(=O)NCC2(OC)CN(C(C(C)N(CC)CC)=O)C2)cncc2ncccc12 Cc1ccc2c(CC(=O)NC(C)(C)CN(C(=O)C#CC3CC3)C)c[nH]c2c1 C(=O)(CC(C)N(C)C(c1sccc1F)=O)NCC1(SCC)CC1 c1(CN2CC(NC(c3cc(C(C)C)[nH]n3)=O)C(F)(F)C2)ccc2nccnc2c1 C=CCC(C(=O)NCCn1ccc(C(N2CCSCC2CO)=O)c1)C(C)C c1(C(=O)NC(COCC)C(=O)NCCCC(O)CO)cccc(F)c1OC c1(C(=O)NCCC2(NC(C3CC(F)C3)=O)CC2)cncc(-c2ccccc2F)c1 c1(CNC(CC(COC)C)=O)ccc2c(c1)CCN(C(=O)CC(C)OC)C2 c1(C(=O)NC2CCCC(NC(CNS(N)(=O)=O)=O)C2)ccn2ccnc2n1 N1(C(c2occ(C(=O)OC)c2)=O)CCC(O)(CCNC(C2(CF)CCC2)=O)CC1 C1(NC(COCCOCC)=O)CCCCC12CCCN(C(C1(N=[N+]=[N-])CC1)=O)C2 N1(C(C(CC=C)C)=O)CCC(C)C(CNC(c2cn(CC(F)F)cn2)=O)C1 c1(CN(CC=C)C(C2CN(c3ccccc3)C(=O)O2)=O)cnc2n(c1=O)CCS2 C1(N(C(CSC)=O)CCSC)CCSC1 c1(C(=O)NCC2C(NC(c3c(C)nc(CC)o3)=O)CC2)n[nH]cc1[N+](=O)[O-] N1(C(C2(CC)CCOC2)=O)CCC2(CCCCN(C(=O)C(=O)NC3CC3)C2)C1 C1(CC=C)(NC(C2CCC(C3CC3)O2)=O)CN(C(c2ccc(COC)o2)=O)C1 c1(CN2CC(CNC(=O)NC(=O)C(Cl)(Cl)Cl)OCC2)cnc(O)c(Cl)c1 c1(-c2cn(CCN(C(C3CC=C(C)CC3)=O)CCO)nn2)ccc(C#N)c(F)c1 N=c1nc2ccc(C(N3CCC4(NC(=O)CCc5ncc[nH]5)CC4C3)=O)cn2[nH]1 c1(CN(C)C)cccc(C(=O)NC(CNC(=O)CSCC2CCCCO2)CO)c1 N1(C(CC(=O)NCC#C)=O)CCCC(C(C)C(=O)Nc2cnn(C(C)C)c2)C1 C1(C(N2C(CNC(C(NC(C)=O)=Cc3cccs3)=O)CC2)=O)CC2(CCOC2)C1 c1(C(=O)NC2C=CCN(C(c3cnn(C)c3C(C)(F)F)=O)C2)cc(N)cc(F)c1 CC1=NOC(C(N2CC3CC2C3NC(=O)CCN2C(=O)CCC2=O)=O)C1C C1(CNC(CCCCC)=O)CCC(F)(CNC(=O)C(c2ccccc2F)O)CC1 C1(N(C(c2cn(CCC)nc2)C(=O)NC(C)(C)C)C)CC2C=CC1C2 Nc1ccc(C(=O)NC2CCCCC2NC(=O)CS(N)(=O)=O)c(F)c1 Cc1nc2c(s1)CC(NC(=O)NC1CC1)CC2.C1(CC2CC2)CNC(=O)N1CC N1(C(c2[nH]c(CC)c(Cl)n2)=O)CCC(C)N(C(c2n[nH]c(C)c2O)=O)CC1 C=CCN=C(NCC(N1CCC(C)CC1)C)N1CCC(C(N2CCCCC2)=O)C1 CC(C)CC(C(=O)NC(C(N1CCC(CCO)CC1)=O)C1(C)CC1)C(C)C CCC(O)C(F)(F)C(=O)N1CC(c2cn(CCOCCOC)nn2)C1 c1(C(C(N2CCC(CN(C)C(c3cccnc3)=O)C2)=O)(C)C)cccc(Cl)c1F N1(C(CNC(C(C)(C)C)=O)=O)CC2(CC(CC(=O)OC(=N)O)C2)C1 c1(OC)c(-c2cc(C(=O)Nc3ncc(C(F)(F)F)cc3N)n[nH]2)cccc1F c1(C(=O)NCC2(NC(c3n(C)cnn3)=O)CC2)ccc(-n2ccnc2)nc1 N1(Cc2cn(Cc3cccc(N)c3)nc2)CCC2(CC1)CC(O)CCO2 c1(C(=O)Nc2cccc(NC(c3n(C)ncc3)=O)c2)cnc(Cl)cc1Cl C(CCC(C)CN1CCCC(C(=O)O)C1)=C(C)C C1(C#N)(C(=O)NC(C)CNC(C2CCCC2c2nncn2C)=O)CC2(CCC2)C1 C1(CNC(C(N2CCC(C)C2)=O)=O)CC(C)(C)CN1C(=O)CC1CCOC1(C)C C1(C(C)(O)CNC(c2cncs2)=O)CCN(C(C2(CC(F)(F)F)CC2)=O)CC1 C(=O)(C(C)S(C)(=O)=O)NC1CCN(C(c2c(C)cco2)=O)C1c1ccccc1 C1(NC(C2CC(C)OC2)=O)CCN(C(c2cc(=O)cc[nH]2)=O)CC1(C)C c1(OC)ccc(C(=O)N(CC(C)NC(c2ccn3c2CCCC3)=O)C)c(N)c1F N1(C(c2ccc(CC)cc2N)=O)CC(C2CN(C(=O)C(c3ccccc3)F)C2)C1 N1(C(c2cc(C)n(C)n2)=O)CC(C(N2CCC(CO)C23CCC3)=O)CC(C)(C)C1 CCS(=O)(=NC(=O)C1(CC=CC)CC12CC2)c1ccc(Br)cc1 Cc1cc(C)c(C(=O)NCCCN(C2CCCC2)C(C2CCCN2C=O)=O)o1 c1(C(N2CCCCC2CCO)C(=O)NC2COC2)cccc2c1CCCC2 c1(N2CCC(SS(CC)=O)CC2)nc(C)cc(=NCC2COC(=O)N2)[nH]1 c1(NC(N(CCCCO)C(C)C)=O)ccnn1CCN(C)C C(C(=O)N(CCC(=O)N1CCC1(C)C(C)C)OC)c1cc(OC)no1 C1(N2CC(c3nnc(OC)s3)C2)C2CCCC(N)C12 C(C(C)(O)CC(=O)NCc1cc(C(=O)NC2CC3CCCC3C2)co1)OC c1(CN2CC(C(=O)NCC=Cc3ccccc3)SCC2)cc(Cl)ccc1Br c1(C(=O)NC2CC(NC(c3cnn(C)c3N)=O)C2)nccn2c(Br)cnc12 C#CC1(C(=O)NC(CNC(=O)COc2ccc(CC#N)cc2)CO)CCOCC1 c1(OC)cc(OC)nc(N(Cc2cn(C)nc2C)CC2(O)CCCNC2)n1 N1(C(CCC(C)NC(=O)CCC(C)(C)[N+](=O)[O-])=O)C2CCC1CN(C)CC2 c1(C(N(CCOC)CCNC(=O)CCCCCF)=O)cnc2n1CC(C)CC2 Cc1nc(-n2cccc2)sc1C(=O)NCC1CCN1C(C1CCOC1)=O C=CCC(CC)C(=O)NCC(C)(C)CC(=O)N1Cc2ncsc2C1 C1(C(=O)NCC(C)NC(C(C)Sc2ncccn2)=O)CC(=O)C1(C)C N1(C(CN(C)CC)=O)CCN(C(c2ccc(OC)cn2)=O)C(CCOC)C1 C1(C(=O)NC2(CNC(CCC(C)O)=O)CC2)CCc2nncn2CC1 C#Cc1ccc(C(N2C(C(=O)Nc3nc(C)ncc3F)CC3CC23)=O)cc1 C(=O)(C(C)CC(=O)N1CCCC(CNC(c2cnccc2COC)=O)CC1)OC N1(C(Cc2cc(C)sc2C)=O)CCCN(C(c2ncn(C(C)C)n2)=O)CC1CO N1(C(C(C)OC2CCOC2)=O)CC(NC(=O)Cc2ccnn2C)C(C)(C)C1 N1(C(C2CC(c3ccccc3)(NC(CC3CN(C)C3)=O)C2)=O)CC2CC1C1CC21 Cc1cccn2c(Br)c(CN3CC4CN(C(=O)CCc5ccsc5)CC34)nc12 c1(C(=O)NC2(CC=C)CN(C(C3OC4CCC3C4)=O)C2)cc(C)cc(F)c1 N1(C(CC(C)C)=O)CC2CCC1C(CNC(=O)Cc1cc(F)cc(Cl)c1)C2 CCC(C#N)(CC)C(=O)NC(C1CCCN(C(C23CSC(C2)C3)=O)C1)C C1(C(C(N2CC3CC3(CNC(C34CC(O)C3C4)=O)C2)=O)O)CCS(=O)(=O)CC1 N1(CC)CCCC(CN(C)CCN2CC(N)C2)C1c1cnn(C)c1 c1(C(N(CC(=O)NCC2(O)CCC(C)C2)C2CCC2)=O)ccn2ccnc2c1 c1(C(C(=O)OC)NC(=O)C(N)CN(C)C)cccc(=O)n1C C(=O)(C(=O)N=c1cc(C)o[nH]1)NCC1CC(NC(C(C2CC2)OC)=O)C1 C1(NC(C(CC#C)C)=O)CC2CCC(C1)N2C(c1cncc(C#N)c1)=O C(=O)(CCC(C)(F)F)N1CCCC(CN(C(COCCN(C)C)=O)C)C1 C1(CC(C)NC(CN2CC(CC)C2)=O)CCCN(C(=O)CC2CCCCCC2)C1 c1(C(N2CCCC2)=O)cnc2c(-c3ccc4c(c3)OCCO4)cnn2c1 N1(CCOC)C2CCC1CN(Cc1n[nH]cc1C(F)(F)F)C2 CC1CCCC(NC(=O)CCC2=CCN(C(=O)C(c3cnn(C)c3)O)CC2)C1C C1(c2ccccc2)(C(=O)N(CC=CC)CC)CC1(C)C.C(CC=O)=C(C)C CC1CC(NC(=O)C(C)OC2CCCCC2)CN(C(c2cc(Cl)ccc2F)=O)C1 c1(NC)cnncc1C(N1CCC(CCC(=O)NCC(C2CCCO2)O)CC1)=O Cn1ccc(C(=O)NCCN2CCC(NC(=O)C(=O)NCCC(N)=O)CC2)cc1=O C1(CNC(CNS(CC)(=O)=O)=O)CN(C(=O)Cc2c(C)n[nH]c2C)CC12CCC2 c1(C(C)C(=O)NCC(C)NC(=O)C(c2cccc(N)c2)O)cccc(F)c1 C(=O)(C#CC(C)(C)C)NC1CN(C(c2c(SCC)cccc2)=O)C(CO)C1 c1(CNCC(c2nnnn2CC2CCOCC2)(C)C)cc(C(N)=O)ns1 C1(C(=O)OCC)CC(N(C(c2ccccc2CC)=O)C(C)C)CCO1 C(=O)(C(CC(C)C)NC(C)=O)NCC1N(C(c2ccc(OC)nn2)=O)CCOC1 CC(C)C(F)C(=O)NC(C)CCCNC(C1(C2CC2)CCC1)=O C1(N(C)C(C2C(c3ccccc3)C2(C)C)=O)CCN(CC2(C)CC=CCC2)CC1 N1(C(c2cnc(C(C)O)s2)=O)C(C)C2CC1C2NC(c1cccs1)=O C1(CNC(C(CC)COC)=O)CN(C(C2(C(C)(F)F)CC2)=O)CC1(F)F Cc1cc(C)n(C(C)C(=O)N(C(C)CNC(c2cnn(C(C)(C)C)c2Cl)=O)C)n1 N1(C(C2CC(C)OC2)=O)Cc2ccc(CNC(=O)C(=O)N=S(C)(C)=O)cc2C1 C1(C(N2CCC(C)(CNC(CC)=O)CC2)=O)CC(C2CCCC2)C1 N12CCc3c(cccc31)C2=O.C(=O)(NNC(=O)c1ccc(I)cc1)C1C(C)C1 c1(CNC(C2CN(Cc3ccc(C4CC4)cc3)CCC2O)=O)cccc(=O)n1O C1(NC(C=CCOC)=O)CCCOC12CCN(C(=O)C#CC(C)C)CC2 C1(C(C)C)C(NC(C23CCN(CC2)C3)=O)CCN1C(c1cccs1)=O c1(-c2ccc(NC(C(C)(C)NCC3CC3)=O)s2)cc(CNS(C)(=O)=O)ccc1F c1(C(=O)NC2C(CNC(C(c3ccc(Cl)cc3)CC)=O)C2)cc(Br)nn1C c1(C(=O)NC2CCC(C)N(C(c3ccc(F)c(F)c3)=O)C2)nc[nH]c2ncnc1-2 CC1CCC(CNCCCOc2ccncc2)CN1 Cc1cnc(Cl)c(C(N2CCOCC(NC(=O)C(C)(C)C3CCCCO3)C2)=O)c1 c1(CC)cc(C(N2CCC(C(=O)N(C)CC3COCCO3)C2)=O)ncn1 N1(C(C=CS(C)=O)=O)CCC2C1CCCN2C(=O)C=Cc1ncc[nH]1 C1(C(N(CC#C)CC=C)=O)CN(C(=O)C(C#N)CC)CCC1(C)C C1(=CC(=O)NCC(CC)NC(=O)C(C)COC)CCC(C)CC1 c1(NC(=O)NCC2(C(=O)OC)CC2(F)F)cccc2cccnc12 CCC(C)(C)C(O)C(=O)NC12CCC(CN(C(c3ccnc4ccsc34)=O)C1)C2 C12(NC(Cc3n(C)ncc3)=O)CCN(C(=O)CCN3CCCCC3)CC1C2 CC1CCc2[nH]nc(C(=O)NC3C4CC3N(C(=O)Cc3nnc(O)s3)C4)c2C1 C1(C(=O)NC(C)CCCCNC(c2cnco2)=O)Cc2cncn2C(=O)N1 N1(C(C(CN(C)C)NC(c2ccnc(O)c2F)=O)=O)CCCC2CN(C)CC12 C12(C(=O)NCC(CO)NC(c3cnn4ccncc34)=O)CCCN1S(=O)(=O)CC2 CC1(C)CC(C)(CO)CN1C(C1CCCCN1C(c1ccc2n[nH]cc2c1)=O)=O C1(C(N(C(CNC(c2cccc(NC)n2)=O)C2CC2)C)=O)CC2CCC1CC2 c1(OCC(=O)NC2C(NC(Cc3cc(C)nn3C)=O)CCC2)c(C)ncnc1C C1(=O)C(CCC(C)c2ccccc2)N2CCC(CC2C)N1.N(CC)(CC)CC C1(N(C)C)CCCC(NCc2ccccc2OCC#N)C1 N1(C(C2(C)C(C)(C)C2)=O)CCC2(CCN(C(=O)Cn3cc(CO)nn3)C2)C1 C(CNC(c1cnn(C(C)C)c1Br)=O)(CC(C)C)NC(CSC)=O c1(N(C(C2CCC(C)NC2=O)=O)CC)nnc(C)c2ccccc12 c1(NC(CN2C(CCC)C(O)CCC2)=O)nc2c(s1)CCCC2 C(=O)(C(F)CCC(C)(C)C)N1CCC(C(C(=O)Nc2c(OC)nsc2)C)C1 c1(C(=O)NC(C(C)C)(C)CNC(=O)CSc2nncn2C)nc2c(s1)COCC2 C1(CCNC(c2ccn(C)c2)=O)CN(C(c2cc(Cl)c[nH]2)=O)CCO1 c1(C(N2CCC3(CCCN3C(=O)C=CC3CC3)C2)=O)cc2ccc(Br)cc2cn1 N1(C(C)C(N2CCCCC2CNC(N)=O)=O)CCC(C2CC(N)CCO2)CC1 C(C(O)CNC(c1cocn1)=O)NC(CSCC(C)C)=O N1(C(CC2ON=C(CC)C2)=O)CCC2CN(C(c3ccc4ncnn4n3)=O)C2C1 C1(NC(Cc2c(C)noc2)=O)C=CCN(C(=O)C(C2CCCCC2)F)C1 C(=O)(C1=CS(=O)CCC1)NCCN(C(c1c(C)ncn1C)=O)C CC1ON=C(C(=O)NCC2CN(C(=O)C(C)(O)C3CCC3)CC2C(F)(F)F)C1C N1(C(c2c(F)ccc(C#C)c2)C(=O)NC(C)CC)CC2(C)CN(C)CC2(C)C1 C1(C(=O)NC(CC)(C)COC)CC=CCC1NC(=O)CCc1ccccc1 c1(C(=O)NC2C(CNC(C=CCOC)=O)C2)ccc(CNS(C)(=O)=O)o1 N1(C(C(CO)NCC(C)C)=O)CCC(C)N(C(C2(CC(F)(F)F)CC2)=O)CC1 N1(C(C(C)NC(CC)=O)=O)CCCC2(NC(c3cc(CC)nn3C)=O)CC2C1 C1(CCNC(CC(=C)C)=O)CCN(C(=O)C(C2CCCC2)OC)CCC1(F)F c1(NC)nc(C)ccc1C(N1CC(CC(C)NC(C2CC(=O)N(O)C2)=O)C1)=O C1(NC(c2cc(OC)c(F)cc2)=O)C2CC3CN(C(c4c[nH]nc4F)=O)C1C3C2 N1(C(CCCNC(C)=O)=O)CCC2CN(C(=O)C(F)C(C)(C)O)CC2CC1 c1(CC(=O)NCC(CC)NC(c2c[nH]ccc2=N)=O)ccc2c[nH]nc2c1 CCCCS(=O)(=O)NC(C)C(=O)NC1COCCC1NC(=O)CC(C)C c1(C(=O)NCC2CC(C(F)(F)F)C2)cccc(Oc2ccc(Cl)cc2)c1 C1(NC(c2cc(CC)on2)=O)CCCCC12CN(C(C1C=CCN1)=O)CCO2 c1(NC(c2ncc(CCCl)s2)=O)ccc2c(c1)CCN(Cc1ccc(O)nc1)C2 CONS(=O)(=O)c1ccc(C(=O)NCC2(CNC(C3CC3F)=O)CCCC2)cc1 C=CCC(C)C(=O)NCCCC1CCN(C(C2OCCOC2C)=O)CC1 c1(CNC(COC)=O)cnn2c1CN(C(c1c(C)cc(O)cc1C)=O)CC2 C1(C(N(CCN(C(C)C)C(c2coc(C(F)F)c2)=O)C)=O)CCC(O)C1 c1(C(=O)NC(C)(C)CNC(=O)C2CC2)nnn(-c2ccc(F)cc2)c1C(F)F C(=O)(CCC(=O)NCCC(C)CCNC(=O)CSCc1nc(C)no1)OCC n1(CCC)cc(C(=O)NCC(O)CN(C(=O)CCOCC(F)(F)F)C)cn1 N1(C(C(C)=C(CC)C)=O)CC(CNC(c2cc(COC)cn2C)=O)C(C)(C)C1 c1(C(=O)NC2C(NC(C3(N(C)C)CCC3)=O)CC2)cnn2cc[nH]c(=O)c12 N1(C(c2cn(CC)nn2)=O)CC2(CCCCN2C(=O)CS(C)(=O)=O)C1 C1(CC)CCCN(C(c2cn(C)nc2OC)=O)C1C(N1CCSC(C)C1)=O N1(C(C(CC)C)=O)C2CCC1C(CNC(c1csc(-c3ccccn3)n1)=O)C2 C12(NC(C3CCC(=O)O3)=O)CC(C1)N(C(C1CCCCC1c1cccnc1)=O)C2 C1(C)(CNC(CNC(CC)=O)=O)CCCN(C(=O)CN2CCCCCC2)C1 N1(C(C(C(C)C)F)=O)CC(N(C)C(C2C3CCCCC23)=O)C2(CC2)C1 C1(CC(=O)N(C)Cc2cccc(F)c2)CN(C(C2(F)CC2(Cl)Cl)=O)CC12CC2 CN1CCCCCC1C(=O)NCC1CCCN(C(c2ccc(N)cn2)=O)CC1 c1(C(C(N2CC(O)(CNC(CCC=C)=O)C2)=O)C)ccc(C#N)cc1 CCC(CNC(=O)CCC1CC1(Cl)Cl)(CC)N=c1nc(-c2ccccc2C)[nH]s1 N1(C(Cn2ccc(=N)[nH]2)=O)CCCC2(CNC(=O)CCCC(F)(F)F)CCCC12 c1(OC)ncc(Cl)cc1C(=O)NCC1(C)CCCN(Cc2cc(C)nc(O)c2)C1 N1(C(c2nccc(OC)c2F)=O)CCC2(C(=O)N(C)C)CCCCC12 N1(C(CCS(C)=O)=O)CCC2(CCCCN(C(c3cnc4[nH]ccc4n3)=O)C2)C1 C(CCCC(CO)NC(=O)CN1CC(C)C1)NC(C(C=C)(C)O)=O C1(CC(N2C(CCNC(CN(CC)C)=O)CCC2)=O)CCC(C)(C)CO1.C(C)(=O)O N1(C(C(c2cccnc2)C)=O)CCC(CNC(C2CCC(=O)N2)=O)C1 C(C(C)(C)C(=O)O)N(C(=O)OC(C)(C)C)C.C(C(C(=O)NCCO)N)OC Cc1ccc(C(C)NC(=O)CCNC(c2csnn2)=O)cn1 C1(c2cn(C3CN(Cc4c(C5CCCC5)nc(C)s4)C3)nn2)CC2CCC1CC2 N(C1CN(C(=O)CS(N)(=O)=O)Cc2ccccc21)C(c1c(OC)ncc(F)c1)=O c1(CNC(=O)NC(CC=C)CN2CC3CCC2C3)c(N)cccc1Cl C1(n2cc(C(COC)(C)O)nn2)CCN(C(c2ccnc(OC(C)=O)c2)=O)CC1 c1(C(=O)NCCC(C)NC(C2(C#N)CCCO2)=O)c[nH]c2cccc([N+](=O)[O-])c12 Nc1cc(C(N2CCN(C(c3coc(CO)c3)=O)C(C(F)(F)F)C2)=O)ccc1F c1(-n2c(C3(NC4CC(C)SC4)CCC(SC)C3)nnn2)cccc([N+](=O)[O-])c1 CC1C(C)N(C(=O)CC23CC(C2)C3)CCN1C(=O)C(C1(O)CCOCC1)(F)F c1(CC(C)N(CC(C(C)C)OCC)C)cc2ccccc2s1 c1(C(=O)NC2CN(C(c3ccc(OC)nn3)=O)CC2C)ccc(Cl)c(OC)c1N N1(C(CCCCOC)=O)Cc2n[nH]cc2C1C(=O)NC1COC2(CCC2)C1 c1(C(N(CC(C)NC(=O)CSC2CCCCO2)C)=O)cc(O)nc(O)c1 N1(C(=O)NC(C(=O)OC)C(C)C)CC2CC(N3CCC(O)C(O)C3)C1C2 c1(C(c2nnnn2CC(F)F)NC2C(C)C2C)ccc(Br)c(Cl)c1F Cc1cc(C#N)ccc1C(=O)NCC(O)CNC(C12CC(C1)C(C(F)(F)F)O2)=O C1(C(=O)NCC(CCOC)NC(c2nccn2C)=O)CCCN(CC(F)(F)F)C1 c1(CC(=O)NCC2(OC)CN(C(=O)Cc3ccccc3Cl)C2)ccc(F)c(Cl)c1 C(=O)(C(CC(N)=O)NC(=O)CC(F)(F)F)NCCNc1c(C2C(C)C2)noc1 C(=O)(C(C#N)C(=O)C=CC1CCCO1)N(CC)CC c1(C(=O)NCC2N(C(c3occ(C)c3C)=O)CCCC2C)ccc2nccn2c1 C1(c2onc(C(C)CCCO)n2)CCN(C(=O)OC(C)(C)C)CC1 Cc1cnc(C(=O)N(C)CCN(C)C(C2CC(=O)C2C)=O)cc1C c1(C(N2CC3C(C(=O)NCC4(O)CCCCC4)(C3)C2)=O)cccn2nccc12 C1(NC(C(CC(N)=O)O)=O)CC2CCC1CN2C(C1CCC(C2CC2)C1)=O C1(CNC(C2CC(C)(F)C2)=O)CCCN(C(c2c[nH]c(=N)s2)=O)CC1 C1(N(C(c2ccc(OC)nc2)=O)C)CC2CC1N(C(C1COCCO1)=O)C2 c1(C(=O)NC(C2CCOC2)CNC(C(CC)CC)=O)cc(C)nc(C(F)F)n1 c1(C(=O)NC(C2N(C(c3c(OC)nsc3)=O)CCC2)C)cccc2oc(O)nc12 C#Cc1ccc(C(N2CCCC(CCNC(=O)CC3CCCC(C)O3)C2)=O)cn1 C1(NC(CC2CC(NC(c3c(C)nncc3)=O)C2)=O)CC2(COCCO2)C1 C(=O)(C1=CCC(F)(F)CC1)NC1(CNC(CC(=O)NCC(F)(F)F)=O)CC1 N1(C(Cc2c(C)n(C)nc2)=O)CCOCC12COCCN(C(=O)C(F)(F)CO)C2 C1(CC)CC(C(C(=O)NC2CCOC2)N(c2nccs2)CCOC(C)=O)C1 N1(C(C2(CS(C)(=O)=O)COC2)=O)CC2(NC(C3CC=CC3)=O)CC1C2 N1(C(c2ccc(CC)nc2C)=O)CC2CCCC2(CNC(=O)CCOC(C)=O)C1 C1(CNC(c2cnn(C3CC3)c2)=O)CCCC1NC(=O)CCN1CCC(F)C1 CC1CN2CCCC2CN1C(=O)C#CC(C)(C)CNC(=O)CC1CC2C=CC1C2 c1(NC(C)=O)ccc(C(=O)NC2CCC(N(C(=O)C=CC3CC3)C)C2)cc1F C1(CCNC(C2CCC=CCC2)=O)CCN(C(C2CCC2(F)F)=O)CC1(F)F CN1CCN(C(C2CCC(O)CN2C)=O)CC1C(N1CC(CC(F)(F)F)C1)=O C1(C(N2CC(CNC(CCCSC)=O)C(C)C2)=O)Cc2ccccc2C1 C(=O)(C(F)(CNC(C1(CC2CC2)CC1)=O)C(C)C)NC(C#C)C(C)C C(=O)(CC(C1CC1)NC(c1cc(Cl)no1)=O)NCCC=CC=C CC1(CNC(C2NC(=O)OC2(C)C)=O)CCCN(C(c2cccnc2)=O)C1 CC1CCCN1CC(=O)NCC1CCN1C(=O)CCSCc1ccccn1 C1(NC(=O)CCN2CCC2)CCN(C(C2(c3cc(Br)ccn3)CC2)=O)CC1 c1(-c2nc(CCCC)nn2C2CCCS(=O)(=O)C2)cc(C)c(C)c(Br)c1 Cc1nn(-c2ccc(F)cc2)c(C)c1CC(=O)NC1CC1NC(=O)C1=CCOC1 C1(C(N2C(CNC(CCC(=O)OCC)=O)CC2)=O)CC(C)CCC1C(C)C c1(CC(N2CCCC(NC(c3scc(C(C)=O)c3)=O)C2)=O)cc(C)ccc1F CCCC(O)(Cn1nnnc1SC)CCC.c12ccc(c(Cl)c1)s2 c1(C(=O)NC2CN(C(=O)C(Cc3ccccc3)C3CC3)C2)cnc(F)c(F)c1 N1(C(CCCC(C)NC(C(C)C(F)F)=O)=O)CCCCCCCC1 C1(C(N2CC(C3N(C(CN(C)C4CC4)=O)CCC3)(O)C2)=O)CCC(C)(C)OC1 C1(NC(C2CC3(CCCC3)CO2)=O)CN(C(C2C=CCC2)=O)C2CCCCC12 C1(C(N(CC(C)CNC(=O)Cc2cccnc2)C)=O)CCCCNC1=O C12(C(N(CC)CC3CC3)=O)CCC(NC(=O)C(c3ccccc3)F)(CC1)C2.C1CC1 c1(OC)cc(Cl)ccc1C1(NC(C2ON=C(C)C2C)=O)CCC1 N1(C(C(CCC)NC(N)=O)=O)CCC(C)(C)C1CNC(=O)CN1CC2CC2C1 C1(NC(COCC(=O)OC)=O)CN(C(=O)C(n2cc(C)cn2)C)CC1OC C1(O)(CN(C(C2(CC#C)CCCC2)=O)C)CCN(C(=O)CCC2CCOC2)CC1 N1(C(C(CC)O)=O)CCC(=CCNC(C2CC2C(=O)OC)=O)CC1 C1(CCC)CN(C(C2COCC2C(F)(F)F)=O)CCN1C(c1nncn1CC)=O c1(C(=O)NC2CCCC(NC(c3nc(N(C)C)oc3)=O)C2)cc2n(n1)CCO2 C#Cc1cc(NC(C2CN(C(=O)CC3CC4CC4C3)CC(C)(C)C2)=O)cc(F)c1 c1(SC)cc(C)c(C(=O)NCC(C2CC2)N(C(=O)CC2NC(=O)NC2=O)C)o1 c1(-c2nc(CCC3CCC(=O)N3)on2)ccc(C(F)F)cc1 c1(CNC(c2sccc2OC2CC2)=O)ccc([N+](=O)[O-])cc1Br C1(NC(CC2C(C)(C)C2)=O)CC2(C1)CC(NC(=O)Cc1ccnnc1O)C2 c1(C(=O)NCC2(OC)CN(C(CCC=C)=O)C2)cnc2sc(C)c(C)n12 CCCN=C(NCC1(C(F)(F)F)CC1)NCC1CC1c1ccccc1OC C(CCC(O)C(=O)NCc1cnc[nH]1)NC(C=CC(C)(C)C)=O C1(C(=O)NC2(CC=C)CN(C(C3(CC)COC3)=O)C2)CCCCC12CC2 N1(C(c2cnc(CC)[nH]2)=O)CC(NC(c2[nH]nnc2-c2ccccc2)=O)C(C)C1 c1(C(N2CCC(C)(CC(=O)Nc3ncco3)CC2)=O)cc(Br)cc([N+](=O)[O-])c1Cl CC1(C(=O)NCC(O)CC2CCCC2)CC(O)CN1C(c1ccsn1)=O N1(C(C(C)OCCC=C)=O)CC(C(=O)NCC(O)CO)C(CC)C1 C1(C)(C(=O)NCC(C2CCC2)OCC)CCN(C(c2ccco2)=O)C1 C=CC(CCC)CC(=O)NC(CC#CC)C(=O)NC(C)C(O)C(F)F Cc1ccc(C(C(=O)Nc2cccc(C3CC3)c2F)N(C2CCC2)C)c(C)c1Br Cc1ccc(C(N2CCOC(CN(C)C(C3CCCN3C3CC3)=O)C2)=O)nc1 c1(C(N(C)CCNC(=O)C(O)Cc2ccccn2)=O)ccc2nnc(O)n2c1 CCCC(CCC)CC(=O)N1CCC(CC(=O)NC(C)C(F)(F)F)C1(C)C C1(C(CO)NC(CSCCC)=O)CCN(C(c2cnc(OC)s2)=O)CC1 CN=S(C)(=O)c1cccc(C(=O)NC2CN(C(=O)C3CCCn4nccc43)C2)c1 Cn1nc2c(c1C(=O)NCc1cc(F)cc(I)c1)CCC2 Cc1nc(CC(=O)NCCN(CC(C)O)C(=O)CC2(C)CC2(Cl)Cl)c(C)s1 c1(C(=O)NCC(CNC(C2(C)C(C)(C)C2)=O)O)cc(N)c(F)c(F)c1Br c1(OC)cccc(C(=O)NC2(C)CC(NC(=O)C(c3ccc(F)cc3)(C)C)C2)n1 c1(OC)c(I)cc(NC(C2CC(O)C(O)C2)=O)cc1I c1(C(=O)NCC(CNC(C=CC(=O)OCCCC)=O)F)cc(Cl)n(C)n1 N1(C(c2cc(C)c(C)nn2)C(=O)NC2CC2)CCc2cccc(C)c21 N1(C(c2nc(SC)sc2)=O)C2CCC1CC(CNC(=O)C(C)C(C)O)C2 c1(C(=O)NCC(C)(C2CC2)NC(C(CC)C2CCOCC2)=O)c(Cl)c(C)nn1C C1(C(N(CC#C)C)=O)CCN(C(=O)CC2COCCO2)C12CC2 C1(NC(c2sc(CC)c(C)c2)=O)CCCCCC1NC(C1CC(C2CC2)=NO1)=O c1(C(=O)NC(C(C)C)C(=O)NC(c2cn[nH]c2)C)ccc2ccoc2c1 C1(COC)CCCN1C(=O)CCC1(C)CN(C(=O)C(c2ccn(C)c2)C)C1 CC1CN(C(=O)CC(C)(C)C)CC(C)N(C(=O)CCN2C(C)CCCC2C)C1 CC(C)CC(O)C(=O)N1CCC12CN(C(=O)C(c1ccc(Cl)cc1)CO)C2 C#CCC(CC(=O)NCCCn1cnnc1C)NC(=O)C(C)(C)C1CCOC1 C(=O)(CCC(=O)c1ccc(O)cc1)N(CCN(C(C(C1CCCC1)OC)=O)C)C N1(C(c2cnc(C(C)O)s2)=O)CC(NC(c2cc(Br)n[nH]2)=O)CC1C N1(C(c2cc(OC)cc(OC)c2)=O)CCC2(CCC(OC)C2)C1.N1(C)CCCC1 C1(C(=O)Nc2cccc(NC(C(CC=CCC)C)=O)c2)CCn2cncc2C1 C(=O)(CCCCCC1OCCO1)NC(C)CN(C1CCSC1)C c1(C(N2C3CN(c4nc(C)cc(C)n4)C(C3)C2)=O)cnc(O)n(C)c1=O c1(C(N2CC(C(C)C)N(C(C3CC(C)(O)C3)=O)CC2)=O)scc2c1CCCC2 N#Cc1cccc(C(N2CC(F)(F)CC2CNC(=O)C(=O)NCC(F)F)=O)c1 Cc1ncc(C(=O)NC2C3CN(C(=O)CC4CS(=O)(=O)C4)CC23)cc1C(F)(F)F c1(N2CC(COC)OCC2)cc(N2CC(C)C(F)C2)nc(C(F)(F)F)n1 c1(C(=O)NCC2(CNc3ncc(C#N)cc3Br)CCC2)nc2ccccn2c1F c1(CC(=O)NCc2ccncc2)ccc(-c2cnn(C3CC3)c2)cc1.C=O CC1C(NC(c2[nH]ccc2CNC(c2ccc(CO)cc2)=O)=O)CCN1C Cc1nccc(N2CCC(NC(=O)C(c3cccc(F)c3)F)CC2)n1 n1(C(CC)C)ccc(=NC(=O)CC2CC(=O)NC2=O)[nH]1 Cc1cc(CC(N2CCCC2CNC(=O)C=C2CCCC2)=O)ccn1 N1(C(c2cc(C)oc2C)=O)CC2(CCCC2NC(=O)C(c2ccc(F)cc2)C)C1 c1(C(=O)NCC(C)CN(C(=O)C(O)c2ccsc2)C)n[nH]cc1Cl N1(C(C2CCCC(C)(C)C2)=O)CCC2(CCC2CNC(c2ccoc2)=O)CC1 C=CCC(CC)C(=O)NC1CC(C(=O)NC2CCCC(C)(C)C2)CC1O N1(C(C2(COC)CCCO2)=O)CC2(C1)CN(C(c1nocc1C)=O)CCO2 N1(C(c2cnc(F)c(F)c2)=O)CCC2CCC(C1)N2c1nc2ccc(Cl)cc2s1 N1(C(c2cccnc2)=O)CCN(C(c2ccc(F)cn2)CNC(C(C)C)=O)CC1 c1(C(N2CCC(NC(CC(C=C)C)=O)C(CO)C2)=O)ccc2snnc2c1 C(C(C)(C)C(=O)N1CCCC(C(C)NC(c2ccncc2C)=O)C1)OC C1(NC(C2C3(CC(NC(CCNC(=O)C=CCl)=O)C3)C2)=O)COC2(CCCC2)C1 CC(=O)CCCC(=O)N1CC2CCC2(NC(=O)Cc2ccn(C3CCCC3)n2)C1 N1(C(=O)C=CBr)CCN(C(C2CC2C(F)(F)F)=O)C(C2CC2)C1 c1(C(=O)NCC2(OC)CN(C(CCCC#CC)=O)C2)ccc2nc(O)cc(O)c2c1 c1(CNC(c2n(CCOC)nnn2)c2ccc(SC)s2)cc(COC)c(C)s1 C1(C(=O)N(C)CCOC2CCC2)(SCC)CCCN1C(=O)C(C(C)C)OC c1(NC(CN(CCCNC(C2(c3cccs3)CC2)=O)CC)=O)c[nH]cc1C c1(C(=O)NCC2(F)CCC(CNC(CC(=C)C)=O)C2)n[nH]c2c1CCSC2 C=C=CC(C)C(=O)N1CC(CC=C)(NC(c2cnn(C(C)C)c2Cl)=O)C1 C1(OC)CC2(C1)CC(C(=O)NCCCOCCNC(C1COCC(C)(C)O1)=O)C2 C=CCC(F)(F)C(=O)NCC(C)NC(=O)CC(C(F)F)c1ccccc1 N1(C(C(C)CO)=O)CCCC12CCN(C(C1(C(F)F)CC(F)(F)C1)=O)C2 C1(NC(c2nnn(CC)c2C)=O)CC2(C1)CN(C(=O)CN(C)S(=O)(=O)N(C)C)C2 C12(C(=O)NCC(CCOC)NC(c3ccnc(OC)n3)=O)CCCN1CC(OC)C2 c1(C(N2CCC(C(C)(C)NC(c3cocn3)=O)C2)=O)ccnc(C(N)=O)c1 C1(n2cnnn2)(C(=O)NC2C(CNC(c3cnc(C4CC4)o3)=O)C2)CCCCC1 c1(NCC(CNC(c2cc(CO)on2)=O)O)cc(-c2cccs2)ncn1 c1(OC)c(C(=O)NCc2cccc(C(=O)NCCc3ncccn3)n2)cnn1C C1(CC(=O)NCCCCCCNC(C2CCCC(=O)N2)=O)CCCC2(CCC2)O1 c1(C(=O)NCC2CCCN(c3ncc(C#N)cc3Br)C2)cccc2oc(O)nc12 N1(C(Cc2n(C)ncc2)=O)CC2CC1CN(C(=O)CC1CCCCCC1)C2 C(=O)(C1CCc2cccnc21)NCCC1C(C)CN(C(=O)CCS(N)(=O)=O)C1 c1(CC(=O)N(C)CC2CCOC2)ccc(Br)cc1Br c1(C(N2C(CN(C(=O)Cc3ccccc3Cl)C)CC(F)C2)=O)csc2nccn12 Cc1csc(C=CC(N2CCC(O)(CNC(=O)C(C)OCC3CC3)C2)=O)n1 C(C1CCN(C(C2CC23CCCCC3)=O)CC1)=CC(=O)NC1(CCC)CCOC1 CCCC(C(O)C(=O)NOCC(F)F)NC(C1CCC(=O)C1)=O N1(C(C(N2CC(C)C2)C)=O)CCC(CCN(C)C(c2cc(F)n[nH]2)=O)CC1 C(=O)(C1=NN(C(C)C(C)C)C(=O)CC1)N(C1CN(C(c2c(C)n[nH]c2C)=O)C1)C CC(C(C)(C)O)N(C(=O)C(C)N(C(=O)CCOC1CCC1)C)C CS(C)(=O)=NS(=O)(=O)NCc1ccc(Br)nc1F c1(OC(CCNC(C(N2CCN(C(CC)C)CC2)=O)=O)=O)ccc(P(C)(C)=O)cc1 C#CCC(CC(F)F)C(=O)N1CCC(CCC(=O)NCCn2ccccc2=O)C1 C1(CNCc2ncc(C)cc2F)COC(C)(C)CN1C(=O)OC(C)(C)C c1(C(N(CCC(C)NC(CCc2cnc(C)o2)=O)C)=O)ccc2nnnn2c1 C1(C(=O)NCCn2cc(CSC)nn2)CC(F)CN1C(c1ncc(F)cn1)=O CC(O)(CNC(=O)CCc1ccoc1)CNC(c1csnc1Cl)=O c1(OCCC(=O)NC(C(C)NC(C2C(CC)C2)=O)C)ccc(OC)cc1 CCCC(C)(CO)NC(=O)CONC(c1cc(CO)c(C)o1)=O c1(CC(=O)NCC(C(C)C)NC(=O)C(C)NC(=O)C(C)(C)C)ccc(Cl)cc1 Cc1cc(C(F)(F)F)nn1CC(=O)C(=O)Cn1cc(C(C)O)nn1.C(C(C)SC)N N1(C(c2c(C)nns2)=O)CCCCC2(CCN(C(=O)C(C3CCOCC3)O)C2)C1 n1(CC)cnc2c(NCc3cc(C)ccn3)[nH]c(=NC(CCO)C(F)F)nc12 c1(CC(=O)NCC2CN(CCO)CC3(CCC3)O2)c[nH]c2ccc([N+](=O)[O-])cc12 CC1(C(N2CC3CC2C3NC(c2ccc3c(c2)COC3)=O)=O)CC(C2CC2)=NO1 C=C(Br)CN=C(NCC1CCCO1)N1CCCC(CC(C)(C)C(N)=O)C1.[nH]1ccnn1 C(C(C)(C)CC(=O)NC1CC1C(=O)NC1CCCN1CCC(C)C)OC C1(CNC(C2C(OCC)C2)=O)(CNC(c2cnn[nH]2)=O)CC12CCC2 C12(CNC(C(CC=C)N(C)C)=O)CCCC1N(C(=O)Cc1cc[nH]c1)CCC2 N1(C(C(C(C)C)SCC)=O)CCC(CNC(C2(C3CCC3)CC2)=O)CC1C c1(NC(=O)C2CC2)cnc2c(c1)CN(C(c1cc(Cl)c(Br)cc1F)=O)CC2 C1(O)(CCNC(C2C(C)(C)CO2)=O)CCN(C(c2cncnc2)=O)CC1 c1(NC(c2cccc(Br)c2)C)cnc(C(F)(F)F)cc1Br C1(NC(=O)CC2CS(=O)(=O)C2)CC12CCOc1ccccc12 c1(CCC)c(C(N2CCC(OCCNC(C3(F)CC3)=O)C2)=O)nnn1C C(=O)(C1CCCc2c1ncn2C)N1CCN(C(CC(C)C2CCCCC2)=O)CC1 c1(C(N(C2CCN(C(C3CC3Cl)=O)CC2)CCO)=O)nccc(Br)c1O C1(NC(C(COC)COC)=O)CCCC12CCN(C(C1CC1F)=O)CC2 c1(C(=O)NC2CCCC(NC(c3coc(O)n3)=O)C2)cnc2ncc(Cl)cn12 N1(C(c2ncn(C(C)C)c2)C(=O)NC2COC2)CCOC(c2cccc(F)c2)C1 C1(CNC(=O)NCCOCC)CC(c2ccc3c(c2)CCO3)=NO1 C1(NC(C(C)(F)F)=O)CCCN(C(=O)CC2=CCCCC2)CC1F C(=O)(CN=c1ccc(C#N)c[nH]1)NCC(CO)NC(C(=Cc1ccco1)C)=O C1(N(C(=O)C(C)C2CC2)CC)CCN(C(=O)CCN2CCCC2=O)CC1 c1(C(=O)NC(C#C)CC)cc(CNC(c2cc[nH]c2)=O)ccn1 C1(SC)COCC1N=c1[nH]c2c(c(=NCCc3c[nH]c(=N)s3)[nH]1)COC2 C1(NC(C(C)CC(N)=O)=O)CC2COCC(C1)C2NC(c1cc(Cl)c(Cl)n1C)=O C1(CNC(C(CCOC)NC(=O)COC(C)(C)C)=O)CC(C)OC(C)C1 C1(NC(c2n(CC#C)ccc2)=O)CC2CCC(C1F)N2C(=O)C(F)CC=C C=CCN=C(NCCCc1cccc2ccccc12)N1CCC2CCCCC2C1 c1(SCC)cc(C(=O)NC2CCCC2NC(=O)CC2CC=CCC2)ccn1 C1(C(=O)NCCC2CCN(C(C(C)=C(C)C)=O)C2)CCCCS1(=O)=O CC1CCc2nc(Cl)nc(N(C3CCN(C(c4cccnc4Cl)=O)C3)C)c2C1 c1(C(CNC(CN(C(=O)Cc2nc(=N)[nH][nH]2)CC)=O)O)cn(C)cn1 C1(NC(=O)OC(C)(C)C)CN(Cc2ncccc2Cl)CCC1C(=O)O N1(C(Cc2cc(C)on2)=O)CC2CCC1C1CN(C(C3C4(CC4)C34CC4)=O)CC21 c1(OC)cc(C(N2CC3CCC2C3)=O)c(NC(=O)C(C)(C)Br)cn1 CC(C)CC(C)(CNC(=O)CCCC1CCC1)NC(=O)C(c1cccc(Cl)c1)C Cc1csc2c(N3CCC4CN(C(=O)C(C)(CO)CO)CC34)ncnc12 N1(C(c2c(NC)scn2)=O)CCC(O)(C(C)CNC(c2nnn(C)c2C)=O)C1 C(CC(O)CNC(c1cnn(C2CCCCC2)c1)=O)NC(C(C)NC(CC)=O)=O Cc1cccc(Br)c1C(C(=O)NC1CC(=O)N(O)C1)NC(=O)Nc1ccsc1C c1(C(=O)NCC(C)N(C)Cc2ccccn2)ccc(F)cn1 N1(C(C2(C)CC2)=O)CC(Nc2ccccc2)C2(CCN(C(=O)C=CCF)CC2)C1 c1(C(N2CCN(C(c3ncc(C)nc3)=O)CC2CO)=O)cnn2c1CCCC2C CCCCCCCCC(=O)NC1CN(C(=O)C(C)(C)CC(=O)OC)CC12CCC2 N1(C(C(CC)n2ccnc2)=O)CCC(O)C(NC(c2nn(C)nc2C)=O)C1 c1(C(=O)NCCCCNC(Cc2cncc(C#N)c2)=O)ccnc2ncsc12 c1(NC(C2CCN(C(c3ccccc3)=O)C2)=O)ccc(OC2CNC2)cc1 c1(C(C(=O)NCCCSC)N(C)CC2CCCSC2)ccc(F)c2ncccc12 CC1CN(C(C2(C)CSC2)=O)CCC1NC(C1(c2ccccc2)CC(F)(F)C1)=O c1(CNC2(NC(=O)OC(C)(C)C)CC2)ncccc1C(F)(F)F CC(=O)CCCC(C)C(=O)NCc1ccoc1C(=O)NOCCC(C)C c1(C(N2CCC(N(C)C(C3SCCS3)=O)C2)=O)ncncc1Br Cc1cc(C2CC2)ncc1C(N1CCCC(F)(CNC(=O)C=CCF)C1)=O c1(C(=O)NCC2(CNC(C3CCC(C)CC3)=O)CC23CCC3)cnc(N)c(Cl)c1 C1(C(=O)N(C)CC2CCCC2(C)C)(CC)CCN(C(C2CC2(F)Cl)=O)CC1 C(CC(=O)NC1CCCC(C(N)=O)C1)(C(F)F)NC(CC1ON=C(CC)C1)=O N1(C(C#CC)=O)CC2CC1C2C(c1ccnnc1C)=O.C1(N2C(=O)C2)CCCCC1 c1(C(=O)NCCC(C)N(C(C=CCOC)=O)C)nnsc1SC CN1CCN(CC(=O)NCc2ccccc2CNc2cc(=O)n(C)cn2)CC1=O c1(CCC)nsc(N)c1C(=O)NCC1CC1NC(=O)C(C)(C)F C1(CC)CCN(C(=O)Cc2sccc2C)C1CNC(C1CCC(=O)N1)=O c1(C(=O)NC)ccc(NC2CC3CCC2N(C(C2CC(=O)N2)=O)C3)c([N+](=O)[O-])c1 CCCC(C(=O)OC)C(=O)N1CC(F)(F)CC1CNC(c1c(C)nn(C)c1C)=O C(=O)(CCCC(=O)NC1CC(F)CN(C(c2cnc(N(C)C)c(Cl)c2)=O)C1)N(C)C C=CCCC(O)CN(C(=O)CC1CCN(C(c2ccccc2)=O)C1)C C1(C(=O)NCC2CCC3(CC3)C2)CCN(C(=O)Cn2cnnc2)C12CC2 C(=O)(CCCN(C)N=O)N1C2C(NC(CC(C(N)=O)NC(C)=O)=O)C(C2)C1 c1(C(N(CCN(C(c2csc(C(F)F)c2)=O)CC)CC)=O)cnc(C(C)C)n1C N1(CC(COC)O)CC2C3CCC(C2C1)N(C(c1coc(S(N)(=O)=O)c1)=O)C3 c1(OC)nc(C(=O)NC2CN(C(C3CC3(F)F)=O)CC2F)cc2ccccc12 CC(C)CC(CNC(c1cc([N+](=O)[O-])c[nH]1)=O)C(=O)NC(C)CC(N)=O c1(C(=O)NC2CCC(NC(CCC(CC)C)=O)C2)cc2cccnc2[nH]1 C1(C(=O)NCCCOCC(C)C)CCN(C(=O)C2=CCOCC2)CC1O C(C)(C(C)SC)N(C(CN(C(=O)CCc1nc[nH]n1)CC)=O)C S(=O)(=O)(CC(C)(C)C#N)N(C(CC#CC)C)Cc1ccccn1 C=CC1(CC(=O)Nc2coc(C3CCC3)n2)CN(C(=O)COCC)C1 c1(OC)cc(C(=O)NC(C)CN(C(=O)C(O)C2CC2)C)ccc1C(N)=O c1(C(N2CCC(C)(NC(=O)CC3CCCO3)CC2)=O)ccc(F)c(F)c1F c1(C(=O)NCC2C(NC(C(C)CN3CCOCC3)=O)CCC2)cc([N+](=O)[O-])c[nH]1 Cc1cc2c(C(=O)NCCCC(C)NC(=O)CCC3CC3C)ccc(C)c2[nH]1 CCC(C)(CO)C(=O)NC1CCCC1n1cc(-c2cnc(F)cc2C)nn1 CCCCC(C)CCC(=O)N1CC(OCCC(N2CCC3CC23)=O)C1 N1(C(C(CCSC)NC(c2c[nH]c(C)c2)=O)=O)C2C=CCC1CCC2 N1(C(c2c(C)ccs2)=O)CCC2C(C1)NC(=O)CN2C(=O)C1=CC(C)CC1 Cc1oc(Br)cc1C(=O)NCC1CC(NC(c2ccncn2)=O)C1 c1(N2CCC(C)C2)cc(S(=O)(=O)N2CCOC(C)(CCO)C2)ccc1C#N c1(CNC(=O)COC(c2ccsc2)=O)ccnn1C1CCOCC1 c1(C(N2CC(C)N(C(C3CC3C3CCC3)=O)CCC2)=O)ccc2ccncc2c1 N1(C(c2c(CC)n[nH]c2)=O)CC2CC1C2C(N1CCC(C)C1C(=O)OC)=O C#CCN(OC)C(=O)C1(F)CCN(C(=O)C(CC)C(=O)OCC)C1 CC1(CNC(c2ccc(Cl)c(F)c2)=O)CN(CC(=O)Nc2ccc(Cl)cc2)CCO1 CCCC(C(=O)NCCOCCOCCNC(=O)CCCC(C)(F)F)C(C)C NC1CCN(C(=O)NCc2ccnc(OC3CCCC3)c2)CC1 C12(NC(C3(C4CC4)CN(C(CC(C)F)=O)C3)=O)CC3CC(CC1C3)C2 c1(CC)nn(C)cc1NC(=O)CC1(C)CCN(C(c2cnco2)=O)C1 C(=O)(C(C(C)CC)C1CC1)N1CC(C=C)(CC(=O)N(CCCCCCO)C)C1 Cc1ccc(C(=O)NCC(C)N(C)C(C2NC(=O)OC2C)=O)cc1C C1(C)(CC)CC(NC(c2cccc(C(N)=O)n2)=O)CN1C(c1cc(C)ncn1)=O N1(C(C(CCC)NC(N)=O)=O)CC(C)OC2(CCN(C(C34CC(C3)C4)=O)CC2)C1 c1(C(=O)NCC2(NC(C3CC(OC)C3)=O)CCCCC2C)ccc2cncn2c1 c1(C(NNC(=O)NCC2OCC(C)(C)OC2)=O)cc2ccccc2o1 N1(C(CSC)=O)CCN(C(c2ccc(C(F)(F)F)c(F)c2C)=O)CC12CCC2 CCC(COC)C(=O)NCC1(F)CCN(C(=O)CCOC(C)=O)C1 C(=O)(C1=CS(=O)CCC1)NC(c1n(CC)ccn1)c1noc(-c2ccccc2)n1 c1(C(N2CCC(CCOC)(NC(c3cn(C)cn3)=O)C2)=O)cccc(C#N)c1F c1(C(N2C(CNC(C3(C)CC3)=O)CC(C(F)(F)F)C2)=O)cc(O)ncc1Br C1(N(C(=O)CC2CN(C)C2)CC)CCN(C(=O)CC2CCCSC2)C1 C1(CC)C(C(=O)NCC(C)CN(C(=O)CCSC(F)(F)F)C)CCN1C c1(C(=O)NC2CN(C(CCOCCOC)=O)CC2O)cc(S(N)(=O)=O)co1 c1(CN(c2ccc(Cl)cc2)CCCC)ccc(-n2cccn2)cc1 C(=O)(C(C)(C)C(C)O)NC1CCN(C(C(F)=CCC)=O)C1 c1(C(=O)NC(CC)CNC(=O)C(CCS(C)=O)N(C)C)cnc2n1CCCCC2 C1(C(N(CC(CCC)O)C)=O)CSCCN1C(c1ccc(CO)s1)=O C1(COC)CN(C(c2cnn(C)c2Cl)=O)CCN1C(=O)CC1(C)CCOCC1 c1(CC(=O)NCC2=CCN(C(=O)C(=O)Cc3cccs3)CC2)cc(F)cc(Cl)c1 C1(C(=O)Nc2c(OC)noc2C)CCCN(C(c2cn(C)ccc2=O)=O)CC1 Cc1ncc(C(N2CCC2CNC(c2ocnc2C(F)(F)F)=O)=O)n1C N1(C(CC(C(=C)C)OCC)=O)Cc2ccccc2C(C)C1 N1(C(C2CCC(C)O2)=O)CC2C(CN(C(=O)CC(C)(F)F)C)C2C1 S(=O)(=O)(c1ccccc1O)N1CCN(CC(CC)(C)CO)CC1 C(CC(F)F)(C(=O)N1CCC(O)CC1C)NC(c1c(C)n(C)cn1)=O c1(C(=O)NC2CCC(CNC(C=C3CCC(C)C3)=O)C2)ccn(O)c(=O)c1 c1(N(C(C)CNC2CCC2)C(C)=O)nc2ccc(F)cc2c(=NC2CCCC2)[nH]1 Cc1cn(CC(N2CCC3CN(C(=O)CSC(F)F)CC23)=O)c(=O)nc1O Cc1ccc(CCC(C)NC(C2CCCCC2c2cccnc2)=O)cc1 C1(C(=O)NCC(COCC)C)(NC(c2cn(CC)nc2C)=O)CCOCC1 C(C(=O)NCC(C)N(C)C(c1sccc1-n1cnnn1)=O)(C(C)C)OCC(C)C C1(CC(N2C(Cn3cc(CNC(C)=O)nn3)CCC2)=O)CCC(C)(C)CO1 c1(C(N(C2CCN(C(c3cccn3C)=O)C2)CC)=O)ccn2ncnc2c1 c1(C(C(=O)OC)NC(c2ccccc2)(C)C)cccc(S(=O)(=O)N(C)CCO)c1 C(CCCCCO)c1cn(C(c2sccc2Br)NC(C2CCCN2)=O)nn1 C1(NC(C(CC=CC)CC)=O)CC2CCCC(C1)N2C(c1cc(CC)n(C)n1)=O N1(C(CCCC)=O)CCC2(COCC(CNC(=O)CC3CCSCC3)O2)C1 N1(C(c2c(C)cnnc2)=O)CCC(C(N2CC(c3ncc[nH]3)C2)=O)C12CC2 CCC(CNC(=O)CCn1ccnc1C)(CC)C(=O)NC(c1nnnn1C)C C1(NC(c2cc(CCC)on2)=O)CC2CC(NC(C3(F)CCOC3)=O)C1C2 N1(C(C2C=CCN2C(=O)C(C2CCOCC2)O)=O)Cc2ncsc2C1 N1(C(C(C2CCOC2)OC)=O)C2CCC1CN(c1cc(=O)n(C)c(=O)n1C)CC2 C=CC(C)(C)CC(=O)N1CCC(NC(c2c[nH]cc2-c2ccc(C)s2)=O)C(F)C1 CC(C)C(C(=O)N1CC2CC1C1CC21)C(C)NC(c1ccc(F)c(F)c1)=O C1(CNC(c2occ(C)c2)=O)CC(NC(=O)CCc2cc(C)on2)CC1O c1(-c2cc(C(N3CC(CNC(CC=CC)=O)C3)=O)no2)ccccc1[N+](=O)[O-] n1(CC(=O)NCCN(CCC)C(c2nc(-c3ccccc3)no2)C)cc(Cl)cn1 C1(CNC(C2(CC)CCOC2)=O)CC(F)(F)CN1C(c1nnccc1C)=O c1(CCC(=O)NCCCN(S(C)(=O)=O)C)nccn1C C=CC1(C(=O)NCC(=O)N(C)O)CCN(C(C2CCC3(CCC3)O2)=O)CC1 C(=O)(C1=CC2CCCCCC12)N1C(CNC(C(c2ccccc2)C)=O)CCCC1 CC1=C(C(=O)N2CC(NC(C3(O)CCCC(C)CC3)=O)C2)C(=O)OC1(C)C c1(OC)c(C(N2CCC(O)(CNC(C3CCC(=O)NC3)=O)C2)=O)cc(Cl)cc1C C1(CC(N2C(Cn3cc(CC(C)(C)OC)nn3)CC2)=O)CCCCN(C(=O)C2CC2)C1 C1(CN(C(c2n(CC#C)ccc2)=O)C)CCCN(C(=O)C(C)C(F)F)C1 CC1CC(CNC(=O)CCc2ccc[nH]2)CN1C(=O)CCC1CC1(C)C c1(C(=O)NC2CC(NC(C3(CC#C)CCOC3)=O)C2)cnc2cc(C)nn2c1C C(C(=O)N1CCN(C(=O)CC2(O)CC2)CC1)(C(C)(C)C)c1n(C)ccn1 c1(C(=O)NC(C(=O)NC(CCCC)COC)Cc2ccoc2)occ2c1CCC2 c1(C(N2CCC(C(C)(C)NC(=O)CSCC(F)(F)F)C2)=O)[nH]ncc1C#N Cc1ncc(Cl)cc1CC(N1CCCC(C)(CNC(C2C(C)(C)C2(F)F)=O)C1)=O c1(NC(c2c(C)[nH]c(C(=O)Nc3cnc(Br)cn3)c2C)=O)ccc(C#N)cc1F CCS(=O)(=O)c1cccc(CC(=O)NC2CC(NC(=O)Cc3ccnn3C)C2)c1 C1(NC(C2C(C)CN(C(c3ccn(C(F)F)n3)=O)CC2)=O)CC2(C1)CC21CCC1 c1(C(N(CC(CN(C(C(C)(C)OC)=O)C)O)C)=O)cc(N)c2ccccc2n1 C1(C(=O)NCc2c(C)n[nH]c2)CCN(C(c2ccc(CF)cc2)=O)C1C N1(C(CSCCC)=O)CCCC(NC(c2sc(F)cc2Cl)=O)C(F)C1 N1(C(CCSC)=O)CC2CCC(N(C)C(C3C4CCCOC34)=O)C2C1 Cc1nc(C(F)(F)F)ccc1C(N1CCCN(C(C2CCS2(=O)=O)=O)CC1)=O Cc1c(C(=O)N(CCCN(C)C(C2CC(F)(F)C2)=O)C)cc(C(C)C)n1C Cc1nc(N2CCC(C)(CNC(=O)C=CC3CCCO3)CC2)c2c[nH]nc2n1 c1(C(=O)NCC2(OC)CCN(C(C3CC(CC)(CC)C3)=O)C2)cc(C)nc(O)n1 C1(CC)CNC(=O)CN1C(=O)C(c1ccoc1)NC(=O)CC(CC)SC C1(N2CC(CNC(C(C)=O)Cc3ccccc3)C2)CCN(C2CCNCC2)CC1 C1(c2n(CC)nnn2)C2Cc3ccc(Br)cc3C12.CN1CCC(c2nnnn2C)C1 C(c1ccoc1)=CC(=O)NCC(CO)NC(c1occc1C1CC1)=O C1(NC(c2c(Cl)ncc(C)c2)=O)CN(c2ncnc(C)c2F)C2CCCCC12 N1(C(CCC(=C)C)=O)CCC(NC(c2cc(Br)cn2C)=O)C(CC)C1 C1(NC(C2(COC)CC2)=O)CCC(O)CN(C(=O)CCN2C(=O)CCC2=O)C1 n1(CC(=O)NC(CC)CC)cc(COCC2CCCO2)nn1 c1(C(=O)NCCCC(C)NC(C23CCC(CO2)C3)=O)cc2ccccc2cc1N c1(C(=O)NC(CC)CN(C(=O)CC(C)(C)SC)C)cc(Cl)cc(Cl)c1 n1(CC)ccc(C(=O)NC2CCC(CCC(=O)NC3(N4CCNC4=O)CC3)C2)n1 N1(C(c2cc(C)n(C(C)C)n2)=O)CC2CC(CNC(C3(C)CCCO3)=O)C2C1 c1(C(N2C(C)CC(CNC(C3CCCCO3)=O)C2)=O)cc(F)c(CO)c(F)c1 c1(C(=O)NC(C(=O)NC(C(=O)NC(C)C)C)c2ccoc2)ccoc1Cl CC(C)(CC(F)C(=O)NCC1CC1(F)F)NC(c1cnc[nH]c1=N)=O Cc1ncc(NC(C23CC(NC(=O)Cc4cccc(C#N)c4)(C2)C3)=O)c(C)c1Br N1(C(=O)CCc2ccco2)CC=CC1CNC(C1(CC2CCCC2)CCCC1)=O c1(C(=O)NCC2C(NC(c3csc(CO)n3)=O)CC2)cc([N+](=O)[O-])n[nH]1 c1(C(=O)NC(CCNC(c2c(CC)nn[nH]2)=O)C(C)C)ccc(F)cc1C n1(CC(=O)NCCCN(C(=O)CCc2cncn2C)CC)ncc(Br)n1 c1(C(=O)NCCCN(C(=O)C(CCSC)OC)CC)nc(C(F)(F)F)ccc1F N1(C(C#CC(C)C)=O)CCC2CCC(NC(C3CC34CC(C)(C)C4)=O)C1C2 CCC(C)(CNC(=O)C(C)Oc1ccccc1)NC(=O)CC1CSCCO1 N1(C(CC(COC)C)=O)CCC(CO)(CNC(c2ccc(C#N)cn2)=O)CC1 CN1CC(O)CC1(C)C(=O)NCC1CC(F)(F)CN1C(=O)CSC(F)(F)F N1(C(C2C(C)OC(C)C2)=O)CC(CO)C2(CCN(C(C3(CCF)CC3)=O)CC2)C1 Cc1cc(C)c(C(N2CCC(NC(c3sccc3C)=O)C(O)C2)=O)c(O)n1 C1(C)(C(=O)NCCCN(C(C2C(C)CCC2)=O)C2CC2)CCC(C)(C)CC1 c1(C(=O)NC2(CNC(c3n(CC(C)C)ncc3)=O)CC2)csc2cncn12 CCCCC(C)C(=O)N(CCN(C(=O)Cc1nnc(S)n1C)C)C(C)C CCCC(C)(O)C(=O)N1CCC(C(=O)NCC2(O)CC(O)C2)C(C)C1 c1(C(=O)NC2CCCN(C(c3c(C)cc(CO)o3)=O)C2C)cc[nH]c2nccc1-2 CC(C)CC(C)(O)C(=O)N(C)CC1CCC(NC(=O)CCc2ncc[nH]2)CC1 Cc1nc(C)c(C(=O)NC2CN(C(=O)CCC3CC3(Cl)Cl)CC2C)c(C)n1 N1(C(=O)CCCc2ccsc2)CC2CN(C(C3CCCC3CF)=O)CC2C1 Cc1c(Cl)ccnc1CNC(c1ccn(CCNC(=O)CNC(=O)C2CC2)c1)=O c1(C(C)O)ccccc1C(N1CC(N2CCN(C(=O)Cn3nccn3)CC2)C1)=O C1(NC(C(C)C)=O)CN(C(=O)CC2CCC2(C)C)CCC1(C)C C(CN=c1ccc(Br)c(S(=O)(=O)N2CCC(n3cncn3)C2)[nH]1)OCCN(C)C N1(C(C(C)(C)OC)=O)CC2(CCOCC2)CC1CNC(=O)C=Cc1ccccn1 N1(C(CCCC(C)=O)=O)CCC2(CC1)CC(C)N(C(c1cnncc1C)=O)C2 N1(C(CCC(CC)NC(c2c(C#N)cnn2C)=O)=O)CC2(CCN(C)CC2)C1 N1(C(=O)C2=CCC2)CCN(C(=O)CC2CCC(O)C2)C(CO)C1 c1(C(=O)NC2C(NC(c3c(C)nc(C(C)(F)F)cc3)=O)C2)cc(Cl)c(F)cc1O C#Cc1cncc(C(N2CCN(C(=O)C(C)n3cncn3)CC2CO)=O)c1 N1(C(C=CCOC)=O)CC(CNC(c2ccccc2NCC(N)=O)=O)CCC1C C#Cc1cc(C(=O)NC2(CC(=O)NCC3=CCN(C(C)=O)CC3)CC2)ccc1C Cc1cc(Br)c(F)cc1C(N1CCOC(CC(=O)NCCC2CCCN2C)C1)=O C1(CC(C)NC(C(C=C)OC)=O)CCN(C(=O)CCOC(C)C)CC1 CC1(CNC(=O)C(F)F)CCN(C(=O)Cc2ccon2)CC1 Cc1nc(-c2c[nH]cc2C(=O)NC2CC(C(C)=O)C2)cs1 C1(NC(c2c(C)noc2)=O)CCN(C(c2cc(C3CCCC3)[nH]n2)=O)CC1F C(CC(C)(C)C(=O)NCC12CC(CN1C(C1(F)CCCCC1)=O)C2)OC C1(C(=O)NCC2(F)CN(C(=O)CCc3ccco3)C2)C(F)(F)C12CC2 C12(NC(c3c(C)nc(C)s3)=O)CCOC(CNC(=O)Cc3cncn3C)(C1)C2 C1(O)(CNC(CC2CC(OC)C2)=O)CCN(C(C2CC(O)CN2C(C)=O)=O)CC1 c1(C(C)C)cc(C(=O)NC(C(=O)NCCCOCCO)C2(C)CC2)no1 c1(C(=O)NCC(CC)NC(=O)C(F)(F)C(O)C(C)C)cnc2c(c1)nc(O)n2C C(=O)(C(C)(C)C(F)c1ccccc1)NCCN(C(c1cn(C)[nH]c1=N)=O)CC1CC1 C1(C(=O)NCCCCNC(C2CC(F)(CO)C2)=O)CCC2(CCC2)OC1 C1(NC(CCn2c(C)cc(C)n2)=O)C(C)CN(C(=O)C=Cc2ncc[nH]2)CC1C C1(C(N2CCC(CC)C2CNC(C2CC(OCC)C2)=O)=O)CCn2ccnc2C1 c1(C(=O)OC)cc(Br)c(C)cc1NC(=O)C(=O)NCC(c1ccc(F)cc1)(C)C CC1(C)CCCC1C(=O)NCC1(F)CC(NC(c2ccc(CO)o2)=O)C1 C12(CC)CC(C(N3CCC(C)C3CNC(=O)CNC(=O)C3CC3)=O)(CO1)C2 C(=O)(C(C)(C)S(C)(=O)=O)NC1CCCC(CN(C(C2(C=C)CCCCC2)=O)C)C1 C1(NC(c2c(Cl)ccc(F)c2F)=O)CCCN(C(c2ccc(O)nn2)=O)CC1F C1(C(=O)NC2CN(C(c3cccn3Cc3ccccc3)=O)C2)(COC)CCOC1 C(CCC(C)(C)C(=O)NCCCC1CC1C)NC(Cc1scc(C)c1)=O C1(CC(N2CCC(CNC(c3c(CC)ncs3)=O)C2)=O)CC(C)(C)CO1 C1(C(N(C(CC)C2CC2)C)=O)CC(F)(F)CN1C(C1CC(F)CN1C)=O C(=O)(C1Cc2ccccc21)NCC1CC(C)N(C(=O)C(F)C(C)(C)O)C1 C1(C)(C(=O)NC2CCCN(CC)C2)CN(C(=O)Cn2cc(C)cn2)CC1C N1(C(C)=O)CCC(NC(=O)C(CCN(C)C)NC(C2(C)CC2(Cl)Cl)=O)CC1 CCC(C(=O)NC1CC(CC(=O)NC2CCCC2CN(C)C)C1)OC C1(C)(CNC(C(C)SC(F)(F)F)=O)CCN(C(=O)CCN2CCOCC2=O)C1 c1(C(N2CCC(NC(c3c(Cl)cccc3Cl)=O)CC2)=O)c(Br)cc(F)c(F)c1F c1(C(C)(C)Cn2cc(CN3C4CSCC3C4)nn2)ncc(Cl)cc1F C(=O)(C(C)CS(C)(=O)=O)N1CCC(O)(CNC(C2(CCC=C)CCCC2)=O)C1 c1(C(=O)NC2C(NC(C=CC)=O)CC2)ccc2n[nH]cc2c1C C1(C(=O)NC23CC(CNC(CNC(CCC)=O)=O)(C2)C3)C2CCOCC12 c1(CNc2c(C(=O)Nc3c(C)ccnc3)scc2)ccc(F)cc1Cl c1(C(N2CCN(C(c3cc(CC)on3)=O)C(C)C2)=O)cc(C)nc2[nH]nc(C)c12 C(CC(F)(F)F)(C(=O)O)N(C(=O)C(O)Cc1cn(CCCO)nn1)C1CCSC1 c1(C(=O)NCCCN(C(C(CC#C)C2CC2)=O)CC)ccn2cccc2c1 C(C(C(=O)NCCCN1CCC1)C(C)(C)C)NC(CC(C(=C)C)OCC)=O N1(C(c2c(C)nc(O)cc2)=O)CC2CC(C1)CN(C(c1cnnn1C1CC1)=O)C2 N1(C(C(C)C(F)F)=O)CC=C(C(C)(C)C(=O)NC2CC(n3ccnn3)C2)C1 C(=O)(C(C1CC1)N(C)C)NCCN(CCO)CC.C12(CCC1)CC(=O)N2C c1(N(C(=O)Cn2cc(C(F)(F)F)cn2)C2COC2)cccc2cc(Br)cnc12 C1(C2CCOCC2)(C(=O)NCC(C)N(C)C(c2cnc(N(C)C)s2)=O)CC1(F)F N1(S(CC2CCCC(C)(C)O2)(=O)=O)CC(C(=O)O)CC12CCOCC2 C1(CNC(C2C(CC)C2)=O)CC2(CCC2)CN1C(C1CN(C(C)=O)CCO1)=O C1(C(=O)OC)COC(CCC(=O)NCCC(C)(C)NC(c2sccc2Cl)=O)C1 Cc1noc(C)c1CNC(N1CCCC1CN(C)C(=O)OC(C)(C)C)=O C1(NC(C=NOC)=O)CC(c2ccc(Br)cc2)N(C(c2cncs2)=O)C1 N1(C(C2N(C(COCCOCC)=O)CCOC2C)=O)C2CCC1CC(O)C2 C1(CC(=O)N(C)CCC2CCC2)CCCN(C(=O)C(C2CCCCC2)O)CC1 Cc1ccccc1OCC(O)CNC(CN1CCCCC1)C(C)C N1(C(C(C)NC(=O)NC)=O)CC(CNC(c2csc(C(C)C)n2)=O)CC1C n1(CC(N2C(C)CC(NC(c3nc(C(C)=O)sc3)=O)C2)=O)cc(S(C)(=O)=O)cn1 C12(C(=O)NC(CC)CN(C)C(c3ccncc3C)=O)CCCCC(OC)(C1)C2 N1(C(C2CCC(C(C)C)CC2)=O)CCC(NC(=O)CSCC(N)=O)C(CO)C1 N1(C(C)C)CCCC(CC(N2CCCC2CNC(=O)C(C)C#N)=O)C1 N1(C(C2N(C)CCC2)=O)CC(CNC(=O)COCC(F)F)C(F)(F)C1 C1(C(=O)NCC(CN(C(c2cc(CC)ncn2)=O)C)(C)C)CC2CCC1CC2 C1(NC(CCSc2ccc(OC)cc2)=O)CCN(C(=O)C2=CCOC2)CC1O n1(CC)nnc(Br)c1CNC(N1CCN(CC2CCC2)CC1)=O c1(CSc2nnc(C)n2Cc2cccc(F)c2)ccc(Cl)c(Cl)c1 CCC(CC)(C(=O)NCC(CNC(C1(C)CC1(F)F)=O)OC)OC C1(NC(C=CC=CC)=O)CN(C(=O)C(C)C)CCC1OC(=O)OC(C)(C)C C12(C(=O)NCc3ccc(C)c(F)c3)CCC(CN(C(C3CCC4(CC4)C3)=O)C1)C2 C12(C(=O)NCC(CNC(=O)CC3(n4cccn4)CC3)F)CCC(O)(CC1)CC2 N1(C(C(=Cc2ncn(C)c2)F)=O)CC(CNC(=O)CC2CCC2(F)F)C(F)(F)C1 c1(CC(=O)NC2(CNC(C3CC(C(=O)OC)C3)=O)CC2)cccc(Cl)c1F CCC(CC)C(C)C(=O)NCC1(OC)CN(C(c2n[nH]c(C(C)(C)C)n2)=O)C1 C1(CNC(=O)CC2CC3(CC3)CO2)CCCCCN1C(=O)C(Cl)=CCl O=C(CCC(=O)c1ccccn1)NCCN(C(=O)C=Cc1ncco1)CC1CC1 C(=O)(CCCC(=O)N1CCOCC(CNC(=O)C(CC)n2cccn2)C1)OC C(C(C)(C)C#CC(=O)NC(C)CCSC)NC(C(C1CC1)SC)=O C1(C(N(CC)Cc2ccoc2)=O)COCCN(C(C2CN3CCC2CC3)=O)C1 N1(C(CN(C)CC)=O)C2CCC1CC(NC(C1COC3COCC13)=O)C2 N1(C(C(CC)O)=O)CCC2CN(C(c3ccc(OC)nc3)=O)CC2CC1 c1(C(N(CC(C)NC(C2CCN(OC)CC2)=O)C)=O)c(N)sc2c1CCSC2 C(=O)(CC(=O)NCCOCCCN(C)C(C1CCC(CC)O1)=O)NCC#C C(=O)(C#CC1CCOC1)NC1C=CCC(C(N2CC(C#N)(F)C2)=O)C1 C=C(C)CC(C(=O)N(C)CC1CCCCN1C(c1sccc1C#N)=O)OC N1(C(C2C(C)OCCC2)=O)CCCN(C(=O)C(C)(C)C2CCOCC2)CC1 c1(OCC(N2C(CCCNC(C(CC)F)=O)CCC2)=O)ccc(F)cc1CO CON1CCC(C(N2CC(NC(=O)C3=CCCSC3)CC2CO)=O)CC1 C1(C(=O)NCC(CNC(=O)Cc2cccs2)CO)CCCC12CC2 C1(N(C(CC(C)SC)=O)CCO)CCN(C(C2(CN3CCOCC3)CC2)=O)CC1 C1(C(=O)Nc2c(CC)nsc2)CN(C(C2(O)CCCCCC2)=O)CC12CC2 c1(OC)ccc(C)cc1CC(N1CCCC(C)C1CNC(c1cc(F)n[nH]1)=O)=O c1(C(=O)NCC2CC(NC(c3c(C)snn3)=O)C2(C)C)cc2n(n1)CCC2 C1(C(=O)NCCOCCC#C)C2CCN(C(=O)CC(C)(C)C#N)CC12 C(C(CO)C(C)(C)C)NC(C1C(CNC(C=C(CC)CC)=O)CCCC1)=O N1(CCO)CCN(C(c2cc(C(=O)NCC3(C)CCOC3)no2)=O)CC1 c1(C(=O)NCC(CC)(C)NC(=O)C(COC)N(C)C)sc2ncccc2c1Cl c1(C(=O)NC2CC(C)(CNC(=O)COC3CCOC3)C2)cc(F)c(F)cc1N c1(CCC(=O)NC(C)CC2CN(C(=O)C(C)N3CCC3)C2)nc(O)n[nH]1 C1(F)(C(N2CC(N(C(c3ccc(C)n3C)=O)C)C(O)C2)=O)CC12CCCCC2 c1(N2CCN(CCOC)CC2)nc(NCCN2CC=CC2)c2ccsc2n1 N1(C(C(CC)NC(C)=O)=O)CCC(C2OCCCC2NC(C2OCCO2)=O)CC1 N1(C(C(CC#C)NC(=O)Cc2ccc(C)cc2)=O)CCCCCCC1 CC1(C)CCN(C(c2ncccc2N)=O)CC1C(N1CCC(F)(F)C(F)C1)=O C(C)(C)(CC(=O)N1CCCCC1CCCNC(=O)Cc1cncc(C)c1)OC C1(CNC(C(=O)NC2(CCOC)CC2)=O)CCNC2(CCC2)C1 c1(C(C(C)NC(C2NCCCC2c2ccccc2)=O)O)ccc2c(c1)OCO2 N1(C(C=Cc2ccc(C)s2)=O)CC(NC(=O)CN(C)C(C)C)C(C2CC2)C1 Cc1ccc(C(C(=O)NCC(C(C)C)NC(=O)Cc2cnccc2Cl)C2CC2)cc1 c1(-c2cn(C3C(SC)CN(C(=O)Nc4ccccc4F)C3)nn2)cccc(F)c1Br C1(NC(C2(CC#C)CCOC2)=O)CCN(C(=O)CCc2csc(C)n2)CC1C N1(C(CCn2ccc(C)n2)=O)CC2CC2(CNC(=O)CCc2ccn(C)n2)C1 c1(C(=O)NC2CN(CCC)C2)sc(S(N)(=O)=O)cc1C N1(C(C(C)NC(=O)NC)=O)CC2CCCC(NC(c3coc(Cl)c3)=O)C2C1 C1(CC(=O)N(CCCN(C)C(N)=O)C)CCN(C(=O)C(F)=CC2CC2)C1 CON1CCC(CC(=O)NCC2CN(C(=O)C(C)(F)CC3CCCC3)C2)CC1 N1(c2ccnc(C(CC)C)n2)CCC(NC(=O)C(CO)NC(N)=O)C2(CCC2)C1 C(=O)(C(C)(C)CC(F)(F)F)NCC(CC)NC(=O)CC1CCC2(CCC2)O1 CC1CCC(NC(=O)CCC2CC2(Cl)Cl)CN1C(=O)Cc1c(Cl)cnn1C CC1(C)CC2(CCN(C(=O)Cn3cn[nH]c3=N)CC2)CO1 C=CCC(CC=C)C(=O)N(C(C)CC(=O)NCC1CCC2(CC1)CC2)C C(CCCCC(=O)Nn1cnnc1C)NC(c1cc(OC)ncn1)=O N1(C(COCCC)=O)CC(C(N2CC(C)C(O)C(C)C2)=O)CC(C)(C)C1 CCCC(=O)NCCC(C)N(C(=O)CCc1cnco1)C C1(CNC(c2ccc(C#C)o2)=O)CC(F)(F)CN1C(=O)CC1(OC)CCOCC1 N1(C2CCN(C(c3cc[nH]c3)=O)C2)CCN(Cc2cc[nH]n2)CC1 N1(C(c2c(C)cc(SC)o2)=O)CCCCC(CNC(=O)Cn2cnnn2)C1 C1(C(=O)OC)CN(Cc2cccnc2CN(CC(C)(C)O)C)CC2CC12 C1(CC=C)(NC(=O)CN2CCC(C)C2)CCN(C(C2(CC)CC2)=O)C1 C1(C(=O)OC)CC12CCN(C(=O)NCCC1(C)CCCC1)C2 Cc1ccc(-n2cc(CN3CCC(C)(NC(=O)C(O)CC(C)C)C3)nn2)c(F)c1 c1(C(C)Nc2c(C)c(NC3CCN(C4CC4)CC3)ncn2)ccc2c(c1)CCC2 c1(NC(N2CCC(c3ccon3)C2)=O)nc2ccc(SC(F)F)cc2s1 NS(=O)(=O)CCCC(=O)NCC(F)CNC(c1cnn(C2CCOC2)n1)=O S(=O)(=O)(c1cccs1)NC(C(=O)NCC1CC(=O)N(C(F)F)C1)Cc1ccccc1 c1(-c2cn(C3CN(C(CSS(C)(=O)=O)=O)C3)nn2)ccc(OCC(F)(F)F)cc1 N1(C(c2c(C)snc2)=O)CCCC(F)(C(=O)NC(CN(C)C)CO)C1 Cc1cc(C(=O)NC2(C#N)CCN(C(c3cc(Br)ccn3)=O)C2)ncc1[N+](=O)[O-] C1(C(=O)NCC2N(C(CCOCCOCC)=O)CCOC2)CCc2c[nH]nc2C1 c1(CCC(=O)NCC2CC(NC(CCCCSC)=O)C2)cnc2ccccc2c1 C12CC(C1(C)C)NC2=O.N1(N(C(=O)CSCC(F)(F)F)C)CC2CC2C1.CC N1(C(CCCCCC)=O)CCOC2(C1)CN(C(=O)CC1CC3COCC13)C2 c1(C(N(C2CCN(C(c3cc(OC)c(C)cc3)=O)C2)C)=O)cc(Cl)cc(C)c1O N1(C(C(CC)Cl)=O)CCC2(CCC2)C(CNC(=O)CC=C(Cl)Cl)C1 c1(CC)nn(C)cc1C(c1nnnn1CCOC)NCCCF c1(C(=O)OCC)ccc(S(=O)(=O)NC(C2CCCOC2)C(=O)OC)cc1C(=O)O C1(CNC(CC=C)=O)N(C(c2c(C)nc(=N)[nH]c2C)=O)CCCC1(C)C c1(C(=O)NCC2C(NC(c3c(C(C)C)occ3)=O)CC2)c(Cl)cnn1C CC1(C)C2CCC1(C(=O)NC1CCN(C(=O)Cc3cn[nH]c3)C1)CC2 CC(C)C(CO)CCNC(=O)C(c1cccnc1)NC(=O)CC1CC(=O)NC1=O c1(C(=O)NC(C2CCN(C(C3CC(C)(C)C3)=O)C2)C)nc(C(F)(F)F)cs1 CC1(C)CC(C)(C(=O)NCCC2CSCCN2C(C2CCCCO2)=O)C1 c1(CCC(N2C(CNC(C3C(CC)CCC3)=O)CC2)=O)ccc(N(C)C)cc1 C1(CNC(=O)C=CC2CCCC2)CCCCN(C(=O)C=Cc2ncc[nH]2)C1 C(=O)(CCC(C)NC(C1CN(C(C)C)C1)=O)NC(CCC=C)C1CC1 C1(CCC)(C(=O)NCC2(CCNC(c3cscc3C)=O)CC2)CCNC1=O CCCCCCC(C)(C)C(=O)NC(C1CCCN1C(c1cnn(C(C)C)n1)=O)C C1(NC(c2ccc3scnc3c2)=O)CCCN(C(C2(F)CC=CC2)=O)CC1F C(C)(C)(CC(=O)Nn1cncn1)N(C(C(C(CC)C)OCC)=O)C C1(NC(C(CN(C)C)NC(CC2(CSC)CC2)=O)=O)CC1C1CC1C C1(CNC(C(=O)NCCOC)=O)CC2CCC1N(C(=O)CCCOC)C2 CCCS(=O)(=O)C(C)C(=O)N1C2CCC1CC(NC(C1CC(=O)NC(=O)N1)=O)C2 N1(C(CS(=O)(=O)NCC)=O)CC(NC(c2c[nH]c(=N)cc2C)=O)CC(F)C1 c1(C(=O)NC2CC(CNC(c3ccc(CCC)cc3)=O)C2)cnn2cccnc12 c1(C(N(CCN(C(C)C)C(C2CC2(F)Cl)=O)C)=O)ccc(F)cc1O c1(NC(CC(C)NC(C2CC(SC)C2)=O)=O)cc(CO)cc(O)c1 c1(OC)ccc2[nH]c(=NC3CCN(C(=O)C(F)C(C)(C)O)CC3C)sc2c1 Cn1c(C(N2CCN(CC(=O)NC3CC(=O)NC3=O)CC2)=O)ccc1C#N C1(C)(CNC(CC2N(CC)CCOC2)=O)CN(C(c2cc(Cl)cs2)=O)C(C)(C)C1 C(=O)(C#CC1(C)CC1)NC1CCCN(C(C(N2CCN(C)CC2)C)=O)C1 c1(C(=O)NC2CC(C)(NC(C(C)OCC)=O)C2)ccc(-n2cnnc2)cc1 C12(NC(C3CCC(N=[N+]=[N-])C3)=O)CCCN(c3ncc(O)cn3)CC1C2 N1(C(C2N(C(CCN(CC)CC)=O)CCC(C)(C)C2)=O)CC(C)OCC(C)(C)C1 c1(C(=O)NC2(CCNC(C(CC=C)C)=O)CCCC2)ccc(OC)c(F)c1O Cc1ccc2[nH]c(C(N3CCC(NC(=O)CC4CCOC4)C(C)C3)=O)cc2c1 Cc1nnc2n1CCN(C(C1(c3cncc(-c4nn[nH]n4)c3)CC1)=O)C2 c1(C(N2CCC(CC(C)NC(C(CC)(C)F)=O)CC2)=O)cc(C)c(O)c(C)c1 C1(C(N(CC(=O)NC2CCCSCC2)C(C)C)=O)Cc2nccn2C1 CCCCC(CC(=O)NCC1CCC(=O)NC1)NC(c1cc(C)nc(O)c1)=O C(=O)(C(CC(C)C(C)(C)C)N(C1CCCC1)CCOC)NCCCCCC n1(CC)cc(C(=O)NC(C(=O)NCC(n2ccnn2)C)C2CC2)cn1 c1(C(N2C(CC)C(=O)NCCC2)=O)cc(O)nc2c1CCCN2 C1(C(N(C)CC2N(C(COCCOC)=O)CC(F)C2)=O)Cc2cc(F)ccc2O1 C1(C(N2CC(NC(C(CC)OCC)=O)C(CO)CC2)=O)CC2(C1)CC(F)(F)C2 C(C)(C(=O)N1CCCC1C(N1CCC(O)C1)=O)(C(C)C)OC O=C1CC(C(=O)NC2C=CC(C(=O)N=c3cc(C(F)(F)F)[nH][nH]3)C2)=CC=N1 Cc1ccn(CC(=O)NC(C)C(c2ccccc2)NC(=O)Cc2cccs2)n1 C1(NC(c2cc(C(N)=O)cc(F)c2)=O)CN(C(c2ccsn2)=O)C2(CCCC2)C1 C(c1cncc(F)c1)=CC(=O)NCCCN(c1ncc(C)cn1)C1CC1 C1(C)(C(=O)NCC(CC)NC(c2cnn(CCO)c2)=O)CC1(C)C C(N=c1ccnc(NC2CC(F)C2)[nH]1)c1n(CC(C)C)ccn1 Cc1cnc2n1CCC(C(=O)N(C)CCN(C)C(c1cnc[nH]c1=N)=O)C2 C(=O)(C(C)(C)CCC#N)NCC12N(C(CN3C(=O)CC(C)(C)O3)=O)CCC1CC2 C(=O)(C1=CCCCCC1)NC1C2CCN(C(CSc3n(C(C)C)cnn3)=O)C21 N1(C(CCC(CC)CC)=O)CCCC2CN(C(=O)C(COC)OC)CC12 CC(C)C(C(=O)N1CCC1CC1CCCC1)Sc1ccccc1 C1(CNC(c2cccc(NC(C)C)c2)=O)CCC(C)CN1C(C1CC2(CC2)C1)=O C=CC(C)CC(=O)NCC1(F)CC(CNC(C2(O)CC(C)(C)C2)=O)C1 c1(C(=O)NC2(C)CC(NC(CC(C)N(C)C)=O)C2)sc(Cl)cc1Cl N1(c2c(C)cnc(C)n2)CCn2ncc(S(C)(=O)=NC(=O)C3C4CCCC34)c2C1 N1(C(C(C)SCCCC)=O)C2CCC1CN(C(=O)C(C)CC(C)(C)C)C2 C#CCCC(O)C(=O)N1CC2C(CN(C)C(c3cc(C(C)C)ccc3F)=O)C2C1 CC1(C)CC(NC(C2CC23CC(O)C3)=O)CN1C(C1CN(C(=O)OC(C)(C)C)C1)=O C1(CC)CN(C(c2cc(COC)cs2)=O)CCC1NC(=O)CCCC#N C(=O)(C1=CCCOC1)NCC1(C(=O)NCCCC=C)CCCC1 C12(C(=O)NC3CCC(CNC(c4scc(OC)c4)=O)C3)CCC(CO)(CC1)C2 c1(CC)cc(C(c2nnnn2C2CCCCC2)NCc2sncc2C)cc(F)c1 C1(NC(CCc2n(C)c3c(n2)cccc3)=O)CCOC2(CCSCC2)C1 CCC(C)C(O)C(C)C(=O)NC(CC)CCC(=O)NC1(C2CCCC2)CC1 C1(CNC(c2c(CC)cc[nH]2)=O)CN(C(c2ccc(SC)s2)=O)CCCO1 N1(C(COCCCCOC)=O)C(C(=O)N(CCCO)C)CCC1C(C)C C1(CNC(CC(C)n2ccnc2)=O)CN(C(=O)CSc2nccn2C)CCC1C C1(CC(=O)NCCc2cc(C(=O)NC(C(=O)N(C)CC)C)no2)CC2CCC1O2 Cc1c(C=CC(=O)NCC2(NC(c3scc(Cl)c3Cl)=O)CC2)cnn1C N1(C(=O)NC2ON=C(C)C2C(C)C)CC2CCOC(=O)C2C1 C#CC1(O)CC(C(=O)N(CC(C)NC(=O)C(c2ccc(F)cc2)CC)C)C1 C1(N(C(c2cccnc2O)=O)CC)CC2CCC(C1)N2C(=O)C(C)NC(N)=O CN1CC(CC(N2CCC(CNC(c3ccc(C(F)F)cc3)=O)CC2)=O)CC1=O C(=O)(C1SCCc2ccccc21)NC1C2CN(C(c3c(C)sc(O)n3)=O)CC21 N1(CCNCCC(C)(c2nnnn2CCCOCC2CC2)N(C)C)CCCCCC1 c1(NC(=O)NC(C2(CC)CN(C(=O)OC(C)(C)C)C2)C)ccc(OC)cn1 c1(C(=O)NCC2(CNC(c3n(CCC)ncc3)=O)CC2)cc(C)nn1CC(F)F c1(CN(C)C)ccc2ccsc2c1.C1(C)(N(C)C(=O)OC(C)(C)C)C(=O)N1 c1(C(N(CCNC(c2cnn(CC)c2C2CC2)=O)C)=O)c(Cl)ccc(F)c1C N1(C(C2(C)CN(C(C3CCC4CC3CO4)=O)C2)=O)CCCC(O)(C2CC2)C1 C1(C(=O)NCC2(CC(=O)N(C(C)CO)CC)CC2)CCC(C)(O)CC1 N1(CC)CCC1C(=O)OC(C)(C)C.C1(=O)CCOC2CN(C2)C(=O)C(C)NCN1 C(C(C)(C)CCN=c1[nH]c(N(C)CC2CCOCC2)nc2cc(C)ccc12)OC CCC(CC)(C(F)(F)F)N1CCCC(CC23CCCC2C3(F)F)C1 C(=O)(C1=C(C)OCCC1)N1CC(NC(CC2CC(CC)OCC2)=O)C(C)(C)C1 CCCCCCC(C)C(=O)NCC(O)CN(C(=O)CC1(C(F)(F)F)CCC1)C C12(C(N3CC(CCOC)N(C(=O)C(O)CC4CC4)CC3)=O)CC(C)(C1)OC2(C)C Cc1ccc(Br)c(C(=O)NC2CCN(C(=O)C3=NOCC3)CC2O)c1 N1(C(c2cn(C)nc2Cl)=O)CCOCC(CNC(C2(C(F)F)CCC2)=O)C1 c1(C(N(C2CCN(C(c3[nH]cc4c3CCCC4)=O)C2)C)=O)cnc2occc2c1 c1(C(N2CC(SC)C(NC(=O)C(C)C)C2)=O)c(F)cc(OC(F)F)cc1F c1(C(=O)NC(c2cn(C)nn2)C(=O)NC(CC)Cn2cncn2)cc[nH]c1C c1(C(=O)NCC2CCC(N(C(CC(C)C)=O)C)CC2)ccc(C(C)(C)C)c(Cl)c1 C1(C(=O)OC)CCN(N2C3CCC2(CO)CC3)C1C1CC1 c1(C(C(C)C)O)ccc(-c2cc(-c3ncccn3)n[nH]2)cc1 N(C1CCOc2ccc(Br)cc21)C(CNCc1ccc(OC)c(OC)c1[N+](=O)[O-])=O Cc1cc(S(N)(=O)=O)oc1C(N1CC2(NC(=O)C3=CCOCC3)CC1C2)=O N1(C(C(C)NC(CC)(C)C)=O)CCC(O)(C(=O)N(CCC(=O)O)CC)CC1 C1(CNC(CCC=CC)=O)CCC2(CCC2)C1NC(c1n[nH]cc1Cl)=O N1(C(CCc2onc(C)n2)=O)CC(C)C(NC(=O)Cc2cncs2)C(C)C1 c1(N2CCC(O)(CNC(C(CCC)OC)=O)C2)nc(Cl)nc(C(=O)OC)c1OC C(=O)(CCC(C)(C)F)NC1(CNC(Cc2ccc(C)cc2)=O)CCOCC1 C(CC(N)=O)(C(=O)NCCC1CCCOC1)NC(CCC1CCC(C)O1)=O C1(CCC#C)CCCN(C(C2(NC(c3cc(F)n(C)n3)=O)CCSC2)=O)C1 Cc1cnncc1C(=O)NC1C=CC(CNC(C2CN(C3CCCCC3)C2)=O)C1 c1(OC)c(CC(=O)NCC(CNC(c2cc(N)nc(Cl)c2)=O)OC)cccc1C Cc1cccc2cc(C(=O)NC3CC(F)CN(C(=O)CCn4cncn4)C3)sc12 C1(NC(C2CC(n3cccn3)C2)=O)CCCC2CN(C(c3cc(Cl)c[nH]3)=O)CC12 C(C(C)(C)CN(C)C)(c1nnnn1NC(C(C1CC1)NC1CCCC1)=O)OCC N1(C(C(C=C=C)C)=O)CC(C)(C)CCC1CNC(c1ncccc1OC(F)F)=O N1(C(c2cccc(OC)n2)=O)CCC2CN(C(=O)CCc3ccc(Cl)s3)CC2C1 CC(C)CCCCCC(=O)NCC1CN(C(=O)C(C)n2cccn2)C2(CCC2)C1 C1(CNC(COCC#C)=O)CC2(CO1)CN(C(=O)C=Cc1ccc(F)c(C)c1)C2 C(C(C)(C)C(C)(C)O)NC(C1(CSC)CN(C(=O)CN2C(=O)CCCC2=O)C1)=O C#CCCCC(=O)N1CC(CCNC(=O)C(=O)NCCCCCCCC)(OC)C1 CC#CCCCC(=O)NCCN(C(C1C(F)(F)C12CC2)=O)CC C1(NC(c2nc(CC(C)C)sc2)=O)CC(CO)N(C(C2CC=CCO2)=O)C1 N(C(=NCCSC)NCCOc1cccc(Cl)c1)C1CCN(C(=O)OCC)C1 c1(C(N(CC(O)CN(C(=O)CS(=O)(=O)NC2CC2)C)C)=O)cccc2c1CCO2 CC1(C)CC(C(=O)NC2(c3cccs3)CC2)CCN1C(=O)CN1CCC(O)CC1 N1(C(C2(OC)CCCC(C)C2)=O)CCn2nc(C(=O)NCc3ccoc3)cc2C1 C(CCCC(=O)N1CC(C)(NC(=O)CCC(O)c2ccccc2)C1)OC C(=O)(C(O)C(C)SC)N1CC(OCC)(CNC(=O)C=Cc2cscn2)C1 c1(C(=O)NC(C2(O)CN(C(CCCOC)=O)C2)C)nc(O)c2ccccc2c1C c1(C(=O)OC)cccc(OCc2ccnn2C(C)CC)c1.C1C(C)O1 N1(C(C2(C=C)CCOCC2)=O)CC(NC(=O)C(CCOC)OC)C2CCCC2C1 CCC(CC)CC(F)C(=O)NC1(COC)CN(C(=O)C(O)c2ccco2)C1 N1(C(=O)Nc2ccc(Cl)c(C(=O)OC)c2F)CCC2(CCCC(C(=O)O)O2)C1 C1(CNC(CC2(COC)CC2)=O)CN(c2nc3ccccc3s2)CCC12CCC2 CCCCCCC(C)CC(=O)N1CC2(CC2)CC1CNC(c1sc(C)cc1C)=O C=CCC(CC)C(=O)NCC1(F)CCN(C(=O)Cc2csc(=N)[nH]2)C1 Cc1c(C(N2CCCC(CC(=O)NCC(C)(O)CN(C)C)CC2)=O)cccc1C#N C1(C(C)NC(C(=O)OC(C)(C)C)=O)CCCN(C(c2ccc(CN(C)C)[nH]2)=O)C1 N1(C(C(C)C)=O)CCN(C(=O)C(C)OCC2CC2)C(c2cccc(F)c2)C1 c1(OC(C(=O)NC2C(NC(c3c(C)cnn3C)=O)C2)C)ccc(F)cc1F c1(C(N2CC3CCN(C(c4ccn(C)n4)=O)C3C2)=O)ccc(Cl)c2cccnc12 Cc1nn(C)c2c(NC(C)C(C)n3cncn3)nc(N3CCCCC(CO)C3)nc12 C(=O)(C1=CC2(CN(C(=O)C3CC3)C2)OC1)N(C(CC#C)C)CC C1(NC(CN(CC)CC)=O)COC2(C1)CN(C(=O)C(C)C=Cc1ccccc1)C2 N1(C(C2C(CC)C2)=O)CC2(C)CN(C(c3ccc(OC)c(O)c3)=O)CC2(C)C1 CC1CCN(C(=O)Cc2cccc(C(N)=O)c2)C(C)C1NC(C1CCSCC1)=O N1(C(c2c(C)n(C(C)C)nn2)=O)C2CCC1C(CNC(C1(F)CCOC1)=O)C2 c1(C(N(C2CCN(C(=O)CCNS(C)(=O)=O)CC2)CC#C)=O)ncncc1Cl N1(C(CCC(CC)CC)=O)CC2CCCN(C(=O)C(O)CC(N)=O)C2C1 c1(CC(C(=O)NCC2OCCC(NC(C=CCCC)=O)C2)C)ccc(Cl)cc1Cl N1(C(C2C(NC(c3ccnc(Cl)c3)=O)C2)=O)CCC2(CC1)CC2CO N1(C(C2=C(C)CC2)=O)CC2CCC(CNC(=O)C(C)NC3CCOC3)C2C1 N1(C(c2c(C)ncs2)=O)CCN(C(c2nccc3cc[nH]c23)=O)C(C)C1C c1(C(=O)NCC2CCCC2C(=O)NCC2CC23CC3(F)F)cc(F)cc(F)c1 c1(C(N(CCCC)CCN(C)C)=O)cn(CCNC(=O)COC)nn1 N1(C(C(C)(C)OC)=O)CCC2(CCC2)C(COCCC(=O)NCC(F)(F)F)C1 CC1COCCN(C(=O)CC2CCN2C(c2ccc(F)c(O)c2)=O)C1 N1(C(COCC(=O)NC)=O)CCC(C(C)NC(=O)Cc2ccn(C)c2)C1 c1(C(=O)NCCC2OCCN(C(C3C(C)OCCC3)=O)C2)ccc2occc2c1 C1(C(=O)NC(CNC(c2c(C)ncn2O)=O)C(C)C)CC(F)(F)C1(F)F c1(CC)noc(CC)c1CC(=O)NC1CC1CNC(c1coc(C(C)C)n1)=O Cc1cc(C(=O)NCC(O)CC(N2CC3(CC3)CC2CO)=O)c[nH]c1=N C(c1cc[nH]n1)=CC(=O)NCCN(C(C1CCN1C1CCCC1)=O)CC c1(OC)cc(NC(C)CCCCNC(C2CCC=CCC2)=O)ncn1 C(=O)(CCCC(CC)NC(=O)CC(CC)SC)N(CC(CCC)C)C C#CCCCCCCNC(C1COCCC1NC(C1(C(=O)C2CC2)CC1)=O)=O CC(C)(C(=O)NC1COC1)C(F)F.C12CCCC1C(C(=O)OC)N2Cc1nccs1 C1(C(N(C2CCN(C(=O)C(=O)NC(C)C)C2)CC)=O)CC(O)C1(C)C c1(C(N(CC(C)O)CCNC(C(F)OC)=O)=O)ccc(CCNS(C)(=O)=O)nc1 C1(CC(=O)NCC2CC(NC(=O)CC3CCN(C4CC4)CC3)C2)NC(=O)NC1=O C1(OC)CC(CO)CN(C(c2ccc(-n3ccc(C(F)(F)F)n3)cc2O)=O)C1 C1(C(=O)NCC(C)(CNC(C2CCC(=O)NC2)=O)OC)CCCCC1N=[N+]=[N-] c1(CCC)[nH]nc(C(=O)Nc2ccc(C(=O)OCC)cc2)c1[N+](=O)[O-] c1(C(=O)NCC2CCC(NC(C(CCC)(C)O)=O)CC2)cccc2nonc12 C1(OC)CC2(C1)CC2NC(c1ccc(CNC(=O)C2=C(Cl)CC2)o1)=O c1(C(=O)NC(c2ccc(O)cc2)CCO)ccc2nccnc2c1 CC(C)CC(C(=O)NC(C)(C)C)NC(=O)CC(C)N(C)C.C1(=O)CN1 N1(C(c2cccc(-c3cnco3)c2)C(=O)NC(C)C)CCC2(COC(C)C2)C1 N1(C(c2nc(OC)oc2)=O)CCN(C(=O)C=CSC)C(C)C1C N1(C(CC=C)=O)CCN(C(=O)Cc2ncc(C)s2)C(c2ccccc2Cl)C1 C1(CN(C(c2cc(COC)on2)C(=O)NCC)C)CCN(CC(F)F)CC1 c1(C(N(CCN(CC)CC)Cc2cccs2)=O)cc2sc(Cl)cc2[nH]1 C#Cc1ccc(C(=O)NCC(C(=O)NC2CC3CCCC3C2)OC)cc1 CC(C)(C)C1=NOC(C(N2CCCC2(C)CNC(=O)CC2C=CCC2)=O)C1 Cc1nc(C(N2CCOCC2CNC(=O)C(c2ccccc2)C)=O)nn1C C=CC(C)(CC)C(=O)NCCC1(CNC(=O)C(C)C(C)(F)F)CC1 n1(CC(N2CCC(C)(NC(C(C)OCCOC)=O)C2)=O)cnc([N+](=O)[O-])c1 Cc1c(C(F)(F)F)cccc1CC(=O)NCC1CCC(C)CN1C(=O)C#CC1CC1 C(=O)(C1=CCN(C(c2c[nH]c3ccccc23)=O)CC1)NCC1([Si](C)(C)C)CC1 CC(C)C(C)C(=O)NCCC(O)C(=O)NCCCN1CCC1 C(=O)(C1CCCc2c[nH]nc21)NCc1cnc(N(CCO)CC)nc1 Cc1ccc(C(N2CC(O)CC2C(=O)NCC2CCCOC2)=O)c(F)c1F Cc1ccc(C(=O)NC2CCCN(Cc3ccnn3C)CC2)c(F)c1F CN1CCN(C(=O)CC2CCSC2)C(C(=O)NCCCN=[N+]=[N-])C1 N1(C(C(C)C2CCCOC2)C(=O)Nc2ccccc2)CCC(C2(C)CC2)C1 C12(NC(c3c(C)cco3)=O)CCC(CC1n1cc(Cn3ccsc3=O)nn1)C2 C1(NC(c2cnn[nH]2)=O)COCCN(C(=O)C(O)Cc2ccccc2Cl)C1 C1(NC(c2cc(Br)c[nH]2)=O)CCN(C(C2CC2(F)F)=O)C1 Cc1ccccc1C(=O)N(C(C)CCNC(=O)C=Cc1nnn(C)n1)C Cc1ccc(NC(=O)C=CC(C)NC(c2ccnn2C(C)C)=O)cc1Cl N1(C(c2ccc(F)c(I)c2)C(=O)NCC(=C)C)CC2(C)CS(=N)(=O)CC2(C)C1 c1(N2CCN(c3ccc(NC(c4ccoc4)=O)cn3)CC2)cc(F)cc(F)c1 c1(C(=O)NCC2C3CN(C(c4ccc(C#C)nc4)=O)CC32)c(C)nc(C)nc1C c1(C(=O)NCCn2nnc(-c3ccccc3)n2)cn2c(n1)SCC2 Cc1nc(N)c2c(C)c(C(=O)NC(C)C(C)NC(=O)CN(C)C(=O)C3CC3)sc2n1 S(=O)(=O)(c1cccc(Cl)c1Cl)NC1C(C#N)CN(C(c2nccs2)=O)C1 N1(C(CN2CC(C)(C)C2)=O)CCN(C(=O)Cc2nc(=N)[nH][nH]2)C2CS(=O)(=O)CC12 C1(NC(CC2(CC=C)CCCC2)=O)CCCN(C(c2c(SC)noc2C)=O)CC1 C1(NC(C(N2CCCC2c2nncn2C)C)=O)COc2cc(Cl)ccc2C1 S(=O)(=O)(c1cccc(NCc2cn[nH]c2)c1)N1C(C#N)CN(C(=O)C2CC2)CC1 C(=O)(C1CCCn2cnnc21)NCCC(C(C)C)NC(C1C(C(F)F)C1(C)C)=O c1cc2c(cc1NC1(c3nnnn3C3CC3)COC3(COC3)C1)OCCC2 CC1(C)CCN(C(=O)C2=CCSC2)C1CNC(C1CC2(CCCO2)C1)=O c1(C(N2CC(NC(C3C(C)SCCC3)=O)C2)=O)ccc2c(n1)CCCN2 C(=O)(C(C)(O)CC)N(C1(CC(=O)N(C)CC2CCN(CC)C2)CC1)C C1(CNC(C(c2ccn(CC)c2)N(C2CCCOC2)CC)=O)CCCC2CC12 N1(CCC(=O)NC2CCC(CCNC(c3ccc(F)s3)=O)C2)CCCCCC1 N1(C(C)C)CCC(CC(N2CCC(C(C)NC(C3CCCCC3)=O)C2)=O)CC1 c1(CCOCC)n[nH]c(=NCCN(C(=O)CCc2ccc(F)cc2Cl)C)s1 c1(C(N(C(CC)CC(=O)NCCC2(O)CCCC2)C)=O)nccc(C)c1N c1(N(C(CNC(C2CCC(C)(CC)O2)=O)C)C)ccc(Br)c(C)c1[N+](=O)[O-] C1(NC(c2c(C(C)C)ocn2)=O)CN(C(=O)C=C2CCOCC2)C2(CCOC2)C1 c1(NC2CCC(SC)C2)nc2c(c(=NCCc3cc(C)n(C)n3)[nH]1)CCCC2 C(CC(C)(C)NC(C1CSCN1C(=O)C=C(C)C(C)(C)C)=O)N(C)C(C1CCC1)=O C1(C(N(CC(C)(C)NC(CC(C)F)=O)C)=O)C2CN(CC(F)(F)F)CC12 c1(C(N2CC3C(CNC(c4cc(C)nc(Cl)c4)=O)(C3)C2)=O)c(F)ccc(F)c1Cl c1(C(N(CCCOCCNC(C(CC(C)C)O)=O)C)=O)sc2nccnc2c1N C(CN=C(NCc1nnnn1C1CCC1)NC1CC1C)N1CC(C)OCC1 c1(C(=O)OC)ccc2nc(NC(=O)NC(CN)C3CC3)sc2c1 N1(C(c2c[nH]c(=NC)o2)=O)CCCC2CN(C(=O)C=CI)CC12 C1(C(N2C(CC)CCC2)=O)CN(C(=O)C(C)(C)N(C)C)CC(C)(C)C1 c1(C(N2CC(C)(NC(=O)C#CC3CCC3)C2)=O)cc2cc[nH]c(=O)c2s1 C1(NC(CC=CC)=O)COCC1NC(=O)C=CBr N1(C(=O)CCSC(F)(F)F)CC2CCC1CN2C(C1CCN1C1CCCC1)=O c1(N2C(C(CSSC)(C)C)CCC2)nc(O)c2cnn(C)c2n1.C1C(=O)N1 C1(CNC(CCC2C(C)=NNC2=O)=O)CC2(CC(NC(=O)C(C)CO)C2)C1 C=CCCCCCCCC(=O)NC1CCC12CCN(C(=O)C=CS(C)=O)CC2 C1(C)(C(N(CC(C)(C)C)CCC#C)=O)CCN(C(=O)CC(C)C=C)CC1 c1(C(N(C)CC2CCNC(=O)C2)=O)cccc(C(=O)C2CC2)c1 N1(C(c2c(CNC(C3(C)ON=C(C)C3)=O)n[nH]c2)=O)CC2(CCC2O)C1 Cn1cc([N+](=O)[O-])cc1C(=O)NCCCNC(c1cc(Cl)ccc1C(F)(F)F)=O c1(C(=O)NC2CCC(C(=O)NC(c3ncnn3C)CC)C2)nc(C)c(C)s1 C1(C(=O)NCCOCCN(C(=O)CO)C)CCCC2CCCN12 C=C(C)CCCC(=O)NCC1CCCCC1NC(=O)Cc1c(F)cccc1F C1(C2CC2)(CNC(=O)C=CC2CCCO2)CCN(C(=O)C2=CCCOC2)C1 c1(C(N2CCOCC(NC(C3(COC)CC3)=O)C2)=O)c(F)ccc(Cl)c1F C(=O)(C(C(C)(C)C)C1CC1)N1CCC(N(C(CC(=O)NCC#C)=O)CCC)C1 C1(C(N2CC(CC(C)NC(c3ncccc3C3CCCC3)=O)C2)=O)CCN(C)C1C N(C(=NCCS(=O)(=O)C(C)C)NCCOc1cccc(F)c1SC)CC Cc1ccc(C(=O)OCC2CN(C3CC3)C(=O)O2)c(P(C)(C)=O)c1 c1(OC)cccc2[nH]cc(CC(=O)NCC(C(C)C)NC(c3scnc3C)=O)c12 CCC1=NOC(CC(N2CCC(CC)C2C(=O)NCC=C(Cl)Cl)=O)C1 Cc1ccc2cc(C(=O)NC(CNC(C3CCC3)=O)C3CCC3)[nH]c2c1 CC1CCC(CNC(=O)C2=COCCC2)N(C(=O)CC23CCC(CC2)C3)C1 CC1OC2(CNC(=O)C(C)Sc3ccccc3)CC1(NC(=O)CNC=O)C2 N1(C(c2ccc(C)s2)=O)CCCC(N(CCO)C(C2(C)COC2)=O)CC1 N1(C(C2N(C)CCCC2)=O)C2CCC1CN(C(=O)C(C)(O)C(C)(C)C)C2 C(C(C)(C)CC(=O)NCCC1(C(=O)O)CCC1)OC C1(C(=O)NC(CC(C)NC(c2c(OC)n[nH]c2)=O)C)CC2(C1)CC(O)C2 c1(C(=O)NCCC(C)NC(=O)CNS(N)(=O)=O)ccc(OC(F)(F)F)nc1 CC1=NS(=O)(=O)NC(C)=C1CC(=O)NC1(CO)CN(C(C2CCC(F)(F)C2)=O)C1 CC1N(C)CCC1(c1nnnn1C1CCC1)NCc1nc(C(F)(F)F)n[nH]1 Cc1nc(O)c2cc(NC(c3cc(Br)c4c(c3)nnn4C)=O)ccc2n1 C1(N2C(COC)CCC2)CCN(C(C)C(C)C)CC1 c1(NC)ccc(Cl)c(C(=O)NC(C)(C)C(C)NC(C2CCC(C)(C)O2)=O)c1 Cc1cc(CC(N2CC(N3CCN(C(C4CCCSC4)=O)CC3)C2)=O)ccc1F C1(NC(CC2N(C)C(=O)CC2)=O)CCC(O)CN(C(=O)Cn2cnccc2=O)C1 N1(C(C(C)=C2CCCC2)=O)CCCC1(C)c1cn(CC2CC(O)C2(C)C)nn1 c1(CC)cnccc1CC(=O)NCC(C)(CO)NC(=O)C(=Cc1c[nH]cn1)F N1(C(C(=O)NCCCC)C2CC2Cl)CCCC(C=O)C1.c1(O)cc(CC)cs1 C1(N(C(c2c(NC)cnnc2)=O)C)CCCCN(C(c2ccc(F)c(O)c2)=O)C1 c1(C(N2C(CC)C(NC(=O)CN3CCCCC3C)CC2)=O)ccc2occc2c1 CCC(C)(C)C(O)C(=O)NC(C)CNC(C1CCC(OC(F)(F)F)C1)=O O(NC(=O)CC(CNC(=O)CC1CCCC12CC2)C1CCC1)C(C)C N1(C(C=CC(C)(C)NC(C2N(C)CC3(CC3)C2)=O)=O)CC2CC3CC2C1C3 C(=O)(C1Cc2ccccc21)N1C(C)CN(C(C2CC2CF)=O)CC1 c1(SCCC(N2CCC(CNC(=O)CN3CC4CC4C3)C2)=O)ccc(Cl)cc1 N1(C(c2cn(CC=C)nc2)=O)CC2CCCC(NC(C3(Cl)CC3)=O)C2C1 c1(C(=O)NC(C(C)NC(c2c(C)cccc2)=O)C(C)C)ccc(C)c(C)c1O c1(C(N2CC(C(=O)Nc3ncccn3)C2)=O)cccc(-c2ccco2)n1 C1(NC(c2ccc(CO)cc2)=O)CN(C(c2ccncc2)=O)C2CC12 C(C(=O)NC1CC(CC(=O)NCCC23CC(CCO2)C3)C1)(C(C)(C)C)OC N1(C(C(c2cccc(C)c2)N)=O)CCNCC2CCCCC12 CN1CCN(C(C2CN(C(C3CCC4(CC3)CC4)=O)CC2(C)C)=O)CC12CC2 C1(C(=O)NC2C(CNC(c3cc(C(N)=O)[nH]n3)=O)CC2)CC(=O)NC(=O)C1 CC1CCN(C(=O)CCC(F)(F)F)CC1NC(c1ccc(-n2cncn2)nc1)=O CC1CN(C(=O)CC2(C)CCC2)CC1NC(C1CCCN(c2cnccn2)C1)=O C(=O)(CS(=O)(=O)C1CC1)N1C(CNC(C2CC(C#C)(O)C2)=O)C(C)CC1 N1(C(C2(C)CNC(=O)C2)=O)C2CCC1C(F)C(NC(c1cc(CCO)on1)=O)C2 CC1CN(CCN(C(=O)C(C2CCN(C(=O)OC(C)(C)C)CC2)F)C)CCO1 CC12CCCCC1C(=O)NOCc1scc(n1)C(=O)N2.c1(CO)cc(O)ccc1F C1(C(N2CC(CC(C)NC(=O)Cc3c(F)cccc3F)C2)=O)CCC(F)(F)CO1 C1(C(=O)NCC(CC)N(C)C(C)=O)CCN(C(=O)C2CC2)C1(C)C N1(C(c2ccn(CC)c2C)=O)CC=C(CC(=O)N2CCCSCC2C)CC1 c1(C(N2CC3(N(C(C(COC)NC(C)=O)=O)CC3)C2)=O)ccc2cnn(C)c2c1 Cc1cccc(Cl)c1CC(=O)NC1CC(NC(=O)C(C)CC2CC2)C(O)C1 c1(OC)ccc2c(c1)OCC2CC(=O)NC1CCN(CC(F)F)CC1 N#Cc1cccc(NC(=O)CC2CCN(C(c3cc4ccccc4[nH]3)=O)C2)c1Cl c1(NC(C2C(NC(C3(C)CCCO3)=O)C2)=O)ncc(Br)cc1OC(F)(F)F c1(-c2cc(C(=O)NCCC3CN(C(C(C)=C4CC4)=O)C3)on2)ccc(F)cc1 C1(CC#N)(NC(=O)C(c2ccccc2)N2CCCC2)COc2ccccc2C1 c1(C(N2CCN(c3c(C(C)(C)C)cccn3)CC2)=O)ccc([Si](C)(C)C)cc1 C1(C(=O)OC)CC(=O)N(C)C1C(=O)NC(C)CCNC(c1cccc(=S)n1O)=O CCC(C)CCCC(=O)N1CCC(CS(=O)(=O)C(F)(F)F)CC1C(=O)O C(=O)(CCCCC(F)(F)F)N1CCC2(NC(CN3CC(C)(OC)C3)=O)C(CC1)C2 c1(C(N2CCCC(C)(F)C2)C(=O)NC(C(=O)OC)C)cnc2ccccc2c1 c1(C(C(F)F)NC(c2oc(Br)nc2C(F)F)=O)cc(F)ccc1F N1(C(C2OCCN(C(C)C)C2)=O)CCCN(C(c2cscc2Cl)=O)CC1C CC1(C)CCN(C(C2CC2C(F)(F)F)=O)CC1C(N1CCC2(CO)CCCC12)=O C1(C)(C(=O)NC2CC(C)(OC)C2(C)C)CN(C(=O)CC2CC=CCN2C)C(C)(C)C1 C1(CC(=O)NC(c2nc(C)sc2)C)CCCN(C(=O)CCCC2CCCO2)C1 N1(C(Cc2c(C)nn(C)c2)=O)CC2=C(C1)CN(C(C1(NC(C)C)CC1)=O)C2 C1(CC(=O)N(C2CCN(C(c3ncc(Cl)s3)=O)C2)CC)CCCC2CCCCC12 C1(NC(c2c(Cl)cc(C)s2)=O)CN(C(c2coc(C(F)F)n2)=O)C2(CCC2)C1 C1(C(N2CC3CC3C2)=O)CC12CCN(S(=O)(=O)CCn1cnc3ccccc13)CC2 N1(C(CNC(c2c(SC)scc2)=O)=O)CCN(C(=O)Cc2ccn(C)n2)CC1 CC1(C)CCC(C)(C(=O)NCC(C2CC2)NC(=O)CC(O)C(Cl)(Cl)Cl)CC1 S(=O)(=O)(CCC(=O)Nc1cc(Oc2ccccc2)ccn1)NC.C1(C)CO1 C1(C(N2C(C(N3CCC3C3CCC3)=O)CC=CC2)=O)CC2(C1)CC(O)C2 N1(C(C(CC)NC(C)=O)=O)CCC2(CCN(C(c3cc(C)c(C)o3)=O)CC2)C1 C(=O)(CCCCC(=O)OC)N1CC(NC(CCOCC)=O)C(F)C1 Cc1nn(C)c(C)c1C(=O)NC1C2CCC(C2)C1C(=O)NC(C)C(F)(F)F c1(C(C)=O)c[nH]c(C(=O)NC(C)CC(C)NC(=O)C(n2nnnc2C(C)(C)C)C)c1 C1(S(=O)(=O)N2CCCC(C(=O)NCC3CCN(C(C)=O)C3)C2)(CC)CC1 Cc1cn2cc(C(=O)NC3CCC3CNC(=O)C(c3ccc(F)cc3)F)nc2s1 CC1(C(N2CCCC(CC#N)C2)=O)CCN(C(=O)C(O)CO)CC1 N1(C(c2cn[nH]c2)=O)CC2CCC(C1)N2C(=O)Cn1nnc(=O)[nH]1 N1(C(=O)CC2CCN(CC(O)CO)C2)CC2CC(O)C2C1 N1(C(C(C)NC(=O)NC2CCCC2)=O)CCC(CNC(=O)CSC(C)(C)C)CC1 C1(C(N(C2CCN(C(c3ccc(SC)o3)=O)C2)CCC)=O)CCC(CF)CC1 S(=O)(=O)(c1ccc(Br)c(Cl)c1)N1CC(F)CC(C(=O)Nc2ccc(SC)cc2)C1 N#Cc1ccc(Br)c(C(=O)NCC2CC(O)CN2C(=O)CC2CC3CC3C2)c1 CCC(C)(F)C(=O)NC1CC(CCNC(c2cc(C3CCCCC3)[nH]n2)=O)C1 N1(C(CC(COC)C)=O)CC2(CNC(=O)C3CC3)CCC1CC2 N1(C(CC2CCCN(C(c3cnc(C)o3)=O)C2)=O)CCC2(CCC(O)C2)C1 C(=O)(C(CC(C)C)C(C)C)N1C2CC(CNC(C3(OCC)CCC3)=O)C1CC2 N1(CC2CC(c3nn(C)c(=O)n3C)CC2O)CC2CCC1CN2CC(=O)O c1(C(=O)OC)ccc(C(=O)NC2(C(C)C)CCC2)cc1.C12CC1CNC2=O c1(NC23C(CN(C(CC(C)OC)=O)C2)CCC3)nc2c(C)cccc2o1 N1(C(Cc2n[nH]c(=NC)s2)=O)CCC(O)(CNC(=O)C(C2(O)CCCC2)F)CC1 c1(COc2c(NC(CN(CCC)C3CC3)=O)cccn2)ccc2c(c1)OCO2 c1(C(=O)NCC2C(NC(c3cc(C)n(C)c3C)=O)CCC2)cscc1S(C)(=O)=O N1(C(CNC(CC)=O)=O)C2CCC1CN(C(c1ccccc1S(C)(=O)=O)=O)CC2 c1(NC(c2cn(CC(=O)N(CC#C)CCOC)nn2)C)[nH]c(O)nc1C c1(N2CCN(CC(C)(F)F)CC2)[nH]c(=NC2CCSCC2)nc2scnc12 N1(C(C(CC)OCC)=O)CCN(C(C)CNC(C2(CCCF)CC2)=O)CC1 C1(NC(C(COC)(C)OC)=O)CCCCN(C(C2(C)CC2)=O)C1 c1(C(N2CCC(O)(CNC(C(CC)(F)F)=O)CC2)=O)ccc2c(c1)OC(C)(C)C2 c1(CC)cc(C)ccc1NC(C1(CNC(=O)CN2CCC(C)C2)CC1)=O N1(C(Cn2cc(CCOC)nn2)=O)CCOCC1(C)C C(CCC(=O)N1CCCC1CCN(CCOC)CCO)OCCC S(=O)(=O)(c1cnn2cc(Br)cnc12)NC(C(C)C1CCOC1)=O C(=O)(C1=CCCCC1)NC(C(=O)N(CCOCC=C)C)CC1CC1 Cc1ccc(S(N)(=O)=O)cc1C(=O)N(C)CC1CCN(C(C2CCC2)=O)C1 Cc1cc(C2CCC2)ncc1C(=O)NCC1CC(NC(C2COC(=O)N2C)=O)C1 N1(C(C(C=CCCC)O)=O)CCC(CCN(C(=O)CC(O)CN(C)C)C)CC1 N1(C(CCS(C)=O)=O)CCOC2(C1)CN(C(c1ccc(N)cc1Cl)=O)C2 CCCCCC(=O)N(CCCCN(C(=O)C(C)=C(C)C)C)C C1(NC(CCOC(CC(C)C)C)=O)CCCN(C(=O)CC2CCCOC2)C1 N1(C(C2N(C(CC(C=C)(C)O)=O)CC2O)=O)CCOCC(C)(C)C1 C1(C(N2CCC(C)(NC(C)=O)C2)=O)CCN(C(=O)CN2CCC(F)CC2)CC1O c1(C(=O)NCCCC(C)NC(CC(n2c(CC)ncc2)C)=O)coc2c1CSC2 c1(NC(CCC=C)=O)cccc(C(=O)NC2CC(C(=O)Nc3ccccc3)C2)n1 C(=O)(C(C)(F)C(=O)N1CC2CC2(CNC(c2cc(C3CC3)nn2C)=O)C1)OCC c1(CCC(=O)NCCC(C)CCNC(=O)C=CC(C)(C)C)nnc(O)nc1O Cc1sc(O)nc1C(N1CCCC1(C)CNC(=O)C(C)NS(C)(=O)=O)=O N1(C(C=CS(C)=O)=O)CC2(CCN(C(c3ccc4nc[nH]c4n3)=O)C2)C1 C1(CNC(c2cn(CCC)nc2)=O)CCC12CCN(C(=O)C(C)COCC)CC2 CCCCCC(CCCCC)C(=O)N1CCC(C(C)NC(c2nc(Cl)cs2)=O)C1 C(=O)(CCCC(=O)NC(C)(C)CCCNC(=O)C(C)(CC)CO)NCC c1(OC)cc(=O)n(C)cc1C(N1CCCC(CN(C(=O)C(C)C(C)C)C)C1)=O C=CC1(NC(C2CCCCC2CNC(=O)C(C)CSC)=O)CCOCC1 N1(C(C(C)OC)=O)CC2(CCC(NC(=O)C(C)Cc3ccc(F)cc3)CC2)C1 N1(C(CC2(OC)CN(C(C3CC=CCC3C)=O)C2)=O)CCC(CO)(CO)C1 c1(C(c2nnnn2CC(F)(F)F)Nc2ccc(F)nc2)cc2c(cn1)OCCO2 N1(C(C(C=C)(C)O)=O)CCC2(CC1)CC2CNC(c1ccc(OC)cn1)=O c1(C(N2CC(C)C(NC(=O)C(Cl)=CCl)C2)=O)ccc(OC(F)F)nc1Cl c1(CCC)ccc(C(N2CCCC2C(C)NC(c2nnc(C)s2)=O)=O)[nH]1 C1(NC(c2c(C)cccn2)=O)CC2CC(C1)N(C(=O)CCCC(C)(C)C)C2 N1(C(C=COCC)=O)CCN(C(C2CC3CCC3C2)=O)CC1CC Cc1cc(N)c(C)nc1C(=O)N(CCCNC(c1c(C)ncn1C)=O)C(C)C c1(CNC(=NC)NC2CC2C(C)(F)F)ccccc1F C12CCN(C1(C)C)C2=O.C=CCC(CNC(C)=O)NC(=O)C(F)(F)c1cccnc1 C1(C(N2C(CCNC(c3ccc(Cl)nc3)=O)CCC2)=O)Cc2cc(Cl)ccc2O1 Cc1ccc(=NC(=O)C2CCCCN2C(=O)C=Cc2cscn2)[nH]n1 C1(C(=O)NCc2nc(CC)on2)CCN(C(=O)CN2CCOCC2)C1C(C)C c1(C(=O)NC(CC)CN(C(=O)C(C(C)(C)C)N(C)C)C)ccc2oc(=O)oc2c1 C1(C(=O)NC23C(CN(C(C4(C(C)C)CC4)=O)C2)C3)CC2(C1)CC1(CCC1)C2 C1(NC(Cn2ccc(C)n2)=O)COC2(CCCN(C(=O)CCC#N)C2)C1 C1(C(C)(C)C)C(=O)N1.C(C(C)CC(F)(F)F)NOCCOC.C1(C)C(=O)N1C1CC1 N1(C(COC(CC)C)=O)CCC(CNC(=O)CCC(F)F)C(C)C1 C(=O)(C(CC1CCC1)NC(C1CS(=O)(=O)C1)=O)NCC(COC(C)C)O C1(CC(=O)NCc2c(C(=O)NCC(C)(C)N3CCCC3)[nH]cc2)CCC(=O)CC1 Cc1ccc(F)c(CN(C(=O)NC2CCCN(c3nc(O)n[nH]3)C2)C(C)C)c1F c1(OC)cc(CC(=O)NC2CCC2NC(=O)C=Cc2cc[nH]c2)ccc1C c1(NC(C)=O)ccc(Cl)c(C(N2C(C(N3CC4CCCC4C3)=O)CC3CC23)=O)c1 C1(C(=O)NCc2cn(CC)nc2)C=CCCN1C(C1CCC(O)CC1)=O Cc1cc(CCC(N2CCC(N(C)C(C3CC(=O)C3)=O)C2)=O)ccc1Br C1(CNC(CCC=CC)=O)(CNC(C2CC2C2CC2)=O)CC12CCC2 C1(NC(c2nc(C)nn2C)=O)CCC12CN(C(=O)CCc1ccccc1Cl)C2 C(c1ccc2ccccc2n1)=CC(N1CC(C)N(C(=O)CC2CC(F)C2)CC1)=O N1(C(c2ccc(CC)s2)=O)CCCC(C(C)(O)CNC(=O)CN(C)CC)C1 Cc1oc2ccccc2c1C(=O)NC1COCC1NC(C1CCCC1C)=O C1(OC)CC(C(=O)NCCN(C)C(C2(C)CC2(F)F)=O)CC1.c1(SC)ccccc1 C1(CCC)CN(C(c2nocc2C)=O)CC1NC(C1CCCC1)=O N1(C(c2nnc(C(=O)OC)s2)=O)CC2CCC1(C(=O)O)C2 Cc1cc(C(=O)NC(C)C(C)(C)NC(=O)CC(F)F)c2cc(F)ccc2n1 c1(OC(C(N2CC(CCNC(C=CC)=O)(OC)C2)=O)CSC)cc(F)cc(F)c1 C1(NC(C2C(COC)C2)=O)C2COCC1CN(C(c1cncc(O)c1)=O)C2 c1(C(CC)=O)cc(C(N2CCCC2C2CCN(C(C3CCCO3)=O)C2)=O)ccc1F c1(C(N(CC(C)NC(CNC(CCCCC)=O)=O)C)=O)ccc2ncnn2n1 C(CCC(=O)NNC(=O)C(C)(C)CCCCNC(c1cc(Cl)ns1)=O)=C(C)C c1(C(=O)NCC2N(C(C3(C(C)(C)C)CCCC3)=O)CCC2)ccc(Cl)cc1N C1(c2nc(C)on2)CN(C(=O)NCc2ncco2)CCO1 C#Cc1ccc(F)c(C(=O)NCCC2CCC(NC(C3CC(CF)C3)=O)C2)c1 N1(C(c2cccc(OC)n2)=O)CC(CNC(=O)C2=NOC(C)C2)C2(CC2)C1 CCC(CC(=O)NCCCC(C)NC(c1ccc(F)cc1OC)=O)CC(C)C CC(C(F)(F)C(F)(F)F)=CC(=O)N(CC(O)CNC(=O)Cc1c(C)noc1Cl)C C1(C(N(CC(C(=O)NCC(N(OCC)C)=O)(C)C)C)=O)CCCC1C1CC1 c1(NC2(C(=O)Oc3c(C)nsc3)CCC2)ccc(Cl)cc1 c1(C(N2CCC(OC)(CNC(=O)C=C3CCCC3)CC2)=O)nc2c(s1)COCC2 Cc1ccc(C(N2CCC2CNC(C2CN(C)CCO2)=O)=O)cc1C#N C(=O)(C(F)(F)CC(=O)N1CC2CC2(CNC(c2cc(C3CC3)on2)=O)C1)OC N1(C(C(C)OCC)=O)CC(CNC(c2cnc3n2CCC3)=O)CC(C)(C)C1 C(=O)(C1=CCCCC1C)N(CC(C(=O)NCc1nnn(CC)n1)(C)C)C C(CC(=O)NC1CCC(NC(=O)C(C)(C)c2ccn(C)n2)CC1)(C(C)C)OCC c12ccc(cn1)c(=O)[nH]2.N12CCCCC1C2.n1(CCC)cc(-c2nn[nH]n2)cn1 C1(O)(C(C(=O)N(C2CCCNC2=O)C)NC(C2CC(F)(F)C2)=O)CCCCC1 N1(C(C(C2CCCCC2)NC(c2nc[nH]n2)=O)=O)CCCC(O)CC1 c1(OC)nc(C(=O)N(CCCCCCNC(C2CCC(O)C2)=O)C)sc1C c1(OC)cc(NC(=O)C=C2CCN(C(c3cc(Br)cnc3C)=O)CC2)c(Br)cc1F CC(=O)CCCC(C)C(=O)N1CCCOC(CNC(=O)CS(=O)(=O)N(C)C)C1 CC1(C(=O)NC2CN(C(c3ccc(S(N)(=O)=O)nc3)=O)C2)CCOC12CC2(F)F C1(NC(Cn2c(C)ccn2)=O)CCCC(N(C)C(C23CC(CO2)C3)=O)C1 C1(F)(C(=O)NC2CCCC(NC(COC(C)(C)C)=O)C2)CCCCCC1 C1(C(N2CCC(C)C2CNC(C2CCCCN2C)=O)=O)CC2(C1)CC2(F)F C1(C(=O)NC2(C(N(OC)C)=O)CC2)C2CN(C(=O)CC3C=NN(C)C3=O)CC12 Cc1cccc(N)c1C(N1CCC(C)(CNC(C2CC2C2CCC2)=O)CC1)=O C1(C)(CNC(C(C)Cn2ccnc2)=O)COCCN(C(c2cnc(O)n2C)=O)C1 CCC(C)CCC(=O)NC(C1CCN(C(=O)CSc2cccc(C#N)c2)CC1)C c1(C(=O)NCC(CCNC(c2c(COC)cco2)=O)O)ccc(Cl)cc1[N+](=O)[O-] n1(CC(=O)N(CC(CNC(C=C(C)C2CC2)=O)C)C)nc(C)cc1C c1(C(=O)NC2CCC(NC(c3ccc(C#N)cn3)=O)CC2)coc2ccccc12 CC(C)CC(C)(C)CNC(C1CCCCCN1C(C1CCS(=O)CC1)=O)=O c1(C(N2CCN(C(c3cc(CC)no3)=O)C(C(F)F)C2)=O)sc2nccn2c1C N1(C(c2c(C)nn[nH]2)=O)CC2CCCC(NC(=O)CC3(CO)CC3)C2C1 C1(CNC(CSCCC)=O)CCN1C(=O)COCC(C)C C1(NC(CCC#CC)=O)CCCN(C(C2CCCN(c3ccccn3)C2)=O)CC1 C1(NC(c2cc(C)no2)=O)CC2(C1)CN(C(C1(Cl)CC13CCC3)=O)C2 C(=O)(C(C)C(C)(C)C)N1CCN(C(Cn2c(C)ccn2)=O)CC1 C(=O)(C(F)C(F)(F)F)N1C(CC)C(C(=O)NCC2CCC3(CC3)C2)CC1 c1(C(=O)NC2(C3CCCN3C(C3CC4(CSC4)C3)=O)CC2)cc2nc[nH]c2cn1 c1(CC(N2CCN(C(c3nc(C)[nH]n3)=O)CC2)=O)c[nH]c2cccnc12 Cc1nc(C(C)C)ccc1C(N1CCC(C(C)NC(C2(C)CCCS2)=O)CC1)=O C1(C(N2CCC(O)(CNC(c3cnc(S)nc3)=O)C2)=O)SC2C=CC1CC2 C1(C(N2CCC(C(=O)NC)C2)=O)CN(C(c2cccnc2C)=O)CCO1 N1(C(c2c(C)cc(OC)nc2)=O)CC(C)CN(C(=O)CCC(F)(F)F)CC1C Cc1ccc(C(=O)NCC2CCC2NC(=O)CC(C)P(C)(C)=O)c2c1CCCN2 CC(C)C(C(=O)NCC(CC1CC1)C(=O)NCc1cccnc1O)C(C)C C(=O)(C1=C(C2CCOC2)N(CCF)C(=O)NC1c1cc2cccc(Cl)c2o1)OC C1(NC(=O)CCc2nc[nH]n2)C=CC(CC(=O)NC2CC2O)C1 C1(NC(=O)CCn2cc(-c3ccc4c(c3)OCO4)nn2)CCC2(CCC2)CO1 N(C1CCCn2nccc21)C(C(CNC(CCc1n(C)ccn1)=O)(C)C)=O C1(C(CNC(C2CC2C(=O)O)=O)F)CCN(C(C2(N3CCOCC3)CC2)=O)CC1 N1(C(c2sc(CC)c(C)c2)=O)CC2(CCN(C(C3CCCC3OC)=O)C2)C1 CC(C)C(C#N)C(=O)NCC(O)CNC(c1ccccc1OCF)=O C#CCC(C)(C(=O)N1CCCC(OCC)C1)NC(=O)CCc1cnn[nH]1 C1(CC(=O)N(C2CCCC2)CCNC(CC=C)=O)CCC2(CCOCC2)CO1 N1(C(c2ccccc2)=O)CCCCC(Cn2cc(C3CCC=CO3)nn2)C1 c1(CC)nocc1C(C(=O)NCCC#N)N(C)Cc1cnn(CC(C)C)c1 C12(C(=O)NCC3(C)CCN(C(C(CCC)F)=O)C3)CCC(CC1F)C2 Cc1ccc(CN2CCCCC2C(=O)NC2CCOCC2O)cc1 c1(C(C)C)ncc(C(N2CC(CNC(C34CC(C3)C4)=O)C2)=O)s1 N1(C(C)=O)CCCCC1C(=O)NCCC1CCN(C(c2ncoc2C2CC2)=O)C1 C1(CNC(C2C3(CC3)C23CC3)=O)CC2CN(C(C34CCCN3CCC4)=O)CC12 C12CCN(C1(C)C)C(=O)C13CCC2C1C3.C1(OC)CCNC1 C12(CNC(C3(OC)CCC3)=O)CCCC(CN1C(c1ccccc1CC#N)=O)C2 C12(CNC(CCCCC)=O)COCCN1C(=O)CN(C(c1ccns1)=O)C2 C1(C(=O)NC2C(NC(c3c(C(C)C)n(C)nc3)=O)CCC2)CC(S(C)(=O)=O)C1 c1(C(N(CCNC(Cn2nc(C)oc2=O)=O)C2CC2)=O)ccc2c(C)noc2c1 N1(C(Cc2nc(C)sc2C)=O)CCCC(NCc2ccc(F)cc2)CC1 C1(NC(C(C2CCC2)OC)=O)CCN(C(=O)CN(c2ccccc2)C)CC1O CCCCC(C)(F)C(=O)NCCCC1CN(C(C2(n3nccn3)CC2)=O)CCO1 c1(CCC(=O)N(C(C)CCNC(C2CCCCC2)=O)C)ccc(C(N)=O)cc1 C1(C(N(C(C(=O)OCC)CSCc2ccccc2)C)=O)CCN(C)S1(=O)=O C1(NC(C(COCC)NC(=O)Cc2cncnc2)=O)CN(C)CC1C C(C(=O)Nc1cccc(CNC(=O)CN2CSCCSC2)c1)(C(C)C)SC C#CCC(CC(=O)N1CC(O)(COC)C1)NC(C1CC1C(C)(C)C)=O Cn1cc2c(n1)CC(C(N1CC=C(CNC(C3CNC(=O)N3)=O)CC1)=O)CC2 C1(C)(CNC(C(C2CC2)OC)=O)CN(Cc2c(F)cccc2F)CCO1 c1(C(=O)NC2CC(c3cn(-c4ccc(C)cn4)nn3)C2)c(C)nn2cccnc12 C1(C(=O)NCC2C(C(=O)NCC(CCOC)O)CC2)COCCN1C C1(C(=O)NC2CC(NC(C(C)CC3CCCC3)=O)C2)CN(C)CC1C(F)(F)F N1(C(C(C=C=C)C)=O)CC(OC)C(OC)C1CNC(c1ccc(C2CC2)cn1)=O C=C1CC2CC1CC2(c1nnnn1CCOC)NCC1CC=CC1 N1(C(C2C(CC)OCC2)=O)CCN(C(c2cn(C3CCC3)nn2)=O)CC(C)C1 Cc1ncc(C(=O)NCCC2CC(NC(c3ccn(C)n3)=O)C2)[nH]1 N1(C(c2cccc(C(C)C)c2)=O)CC2(NC(=O)C3CC3)CCC1CC2 C(C(CC1CCCC1)C(=O)Nc1ccc(F)cc1)NC(C1CCN(CC)C1)=O Cc1nn(C)c(C)c1C(=O)NC1(C#N)CCN(C(c2cc(Br)ccn2)=O)C1 Cc1ccncc1C(C1CC1)NC(=O)CCn1cc(CC(O)C(C)(C)C)nn1 Cc1cc(NC(C2CC(C)CN2C(c2ncccc2N)=O)=O)c(C)c(C)c1 n1(CC)c(C)cc(C(=O)NCCNC(=O)C(C)Cc2cccc(F)c2)c1C Cc1cnc(N)c(C(=O)NC(C)(CNC(=O)Cc2sccc2C)CO)c1 C1(NC(C(C2(O)CCC2)NC(C=CCC)=O)=O)CCC(=O)NC1(C)C CN1Cc2cc(NC(C3CCCC4CCC3N4)=O)ccc2C1=O C1(C(=O)NCC(=C)F)CCC(C)N(C(c2ccc(=N)[nH]c2)=O)C1 N1(CC(=O)NCc2ccc(C(N3CC(c4nn[nH]n4)C3)=O)o2)CCCCC1=O CC12CCN(C(=O)CC3CCCSC3)C1CN(C(c1cnn3c1SCC3)=O)C2 Cc1cccc(-n2cc(CC3CCN(C(C4(C)C=CCC4)=O)C3)nn2)c1[N+](=O)[O-] Cc1ccccc1.C1(CCN(CCCO)C(=O)Cn2ccnn2)CCCCC1 CCC(C)(COC)C(=O)NCc1csc(CNC(=O)CC(C)(C)C)n1 c1(C(=O)NCCC2CCCCN2c2ncc(O)cn2)cc(F)cc2ccoc12 C1(CC(=O)N(CCCC#C)C)CN(C(C2CC=CCC2)=O)CC1C N1(C(COc2cccc(C#N)c2)=O)CCN(C(c2ccc(Cl)s2)=O)C2CCC12 c1(CNCC)cccc(C(=O)NCCC2CCCO2)c1 n1(CC(=O)NC(C2(O)CCN(C(C(C)=CC)=O)CC2)C)cc(S(C)(=O)=O)cn1 S(=O)(=O)(c1ccc(Cl)cn1)NCC(c1ccco1)(OC)OC N1(C(C(=Cc2ccco2)C)=O)CC(C)N(C(=O)CN2CCOCC2)CC1C C1(NC(CCCc2ccc(C)s2)=O)CCCN(C(=O)CCC2CCCN2C)C1 C1(NC(c2c(C(=O)OC)cco2)=O)CCOC(C(=O)NCCCC2CCCC2)C1 C1(CCC(=O)NCC2C(C(=O)NC(CCC)C)C2)CCC(=O)C1 C1(NC(C2(C(C)C)CCC2)=O)CCN(C(c2cccnc2Br)=O)CC1F N1(C(Cc2cn(CC)nc2)=O)CCN(C)CC1CNC(=O)C(C)CC1CC1 c1(NC2CC3CN(C(CCCOCC)=O)CC32)nnc2c(c1C(F)(F)F)CCC2 c1(C(=O)NCCN(C(=O)NCC)C)cc2c(cc1C(=O)OC(C)(C)C)CCC2 C1(C(N2CC(C)C(CO)CC2)=O)CCCN1NC(=O)C1(C)CCOCC1 C(C(=O)NC1CC(CCNC(C2(CO)COC2)=O)C1)(C(C)C)c1cnc(C)s1 CC1CN2CCN1CC2C(=O)NC1CC(O)C(O)C1O C(CNC(=O)C(Cn1cccn1)NC(c1n[nH]cc1Cl)=O)(C(C)(C)C)OC c1(C(=O)NCCCC(C)NC(C2(C#N)CCC2)=O)cnn2cccnc12 c1(C(N2CC(C)C(NC(=O)C(C)(C)CC#N)CC2)=O)cccc2c1CNC2=O C1(CC(=O)NC)CCCCC12CC2.C1C(=O)N(CC(C)O)CCN1CC c1(Cn2ncc(NS(=O)(=O)C(F)(F)F)c2)ccc2nonc2c1 C1(N(C(C(C2CCCC2)SC)=O)CCO)CCN(C(=O)CCNC2CC2)C1 C1(C(=O)N(CC(C)Nc2ccc(OC(F)F)cn2)C)(CC)CCNC1=O N1(C(C2(C)CC3CCC2C3)=O)CCC2(CCCN(C(=O)CCP(C)(C)=O)C2)C1 c1(C(=O)NCC2(NC(CCCCC)=O)CCOC2)cc(F)cc2nccnc12 N1(C(COCCC=C)=O)CCC(NC(=O)C(C)(C)CNC(C)=O)C(O)C1 N1(C(C2(CC#C)CCN(C(=O)C(C)OC(C)=O)C2)=O)CC2OCC(CO)C2C1 c1(NC(=O)NC(C)C(C)n2cccn2)cc(C(N)=O)ccn1 C1(CNC(Cc2c(C)noc2C)=O)CCN(C(c2ccc(O)c(F)c2)=O)CC1C C(c1ccc2c(c1)OCO2)=CC(=O)NCCCOCCNC(C(C)CS(C)=O)=O CCC(C(=O)NC1CC2CN(C(=O)C(c3ccc(F)cc3)C)CC12)C(C)O N1(CN(C)Cc2cccc(C(C)C)c2)CC2(C1)CN(CCc1ncccc1F)C2 C1(CCC)CCCC1C(=O)NC1(C(=O)N(C)Cc2occc2C)CSC1 c1(C(C(=O)NCC2CCN(C(C3(COC)CCC3)=O)C2)=O)nn(C)cc1Br C(N=c1nc2[nH][nH]cc-2c(O)n1)C1CC(NC(c2ccc(OC)nc2)=O)C1 N1(C(C2C(C)=CCS2)=O)CC=CC1(C)C(=O)N(C)CC1CC(F)C1 Cc1onc(CC(N2CC(NC(C3(COC(C)C)CC3)=O)CC(C)C2)=O)c1C#N C(c1ccc(Cl)cc1F)=CC(N1C(C(=O)OCC(=O)NC)CC(C)C1)=O C(c1cn(C)nn1)=C(C(=O)NCCCCNC(CN(C(=O)OC(C)(C)C)CC)=O)F CCC(C)CC(C)C(=O)N1CCN(C(C23CCCN2CCC3)=O)C2(CC2)C1 N1(C(CCCCC#N)=O)CCN(C(C2CCCCN2C(N)=O)=O)CC(CO)C1 C1(NC(C(CCC)N(C)C)=O)CCC2CN(C(c3cncnc3C)=O)CC2C1 c1(C(=O)NCC(c2n(C)ncc2)O)ccc(S(=O)(=O)N2CCOCC2)o1 c1(CC)cccc(C(=O)N(CCCN(C(=O)CCN2CCCOCC2)C)C)c1N N1(C(c2nnsc2CC)=O)CCC(C)C(N(C(=O)COc2ccc(C)cc2)C)C1 N(C)(C1c2ccccc2CC1O)C(=O)N(c1n(CC(F)(F)F)nc(C)c1[N+](=O)[O-])CC c1(CC(N2CC(C)N(C(C3CC(C)(O)C3)=O)CC2)=O)ccc2nn(C)cc2c1 c1(C(=O)NC(C2CCN(C(c3csc(=N)[nH]3)=O)C2)C)cnn2c1CCC2 c1(CC(C)C)ccc(CCCNC(C2CCCOC2)C)cc1 c1(C(=O)OCC)cc(=NC(=O)c2nc(Nc3ccc(OC)c(C)c3F)cs2)[nH][nH]1 N1(CC(=O)NC)CCC2(CCN(C(c3ccc(-c4noc(C)n4)cc3)=O)C2)C1 c1(C(N(CCN(C(CSCC)=O)C(C)C)C)=O)cc(-c2ccncc2)ccn1 C#CCC(O)C(=O)NCC(CC)NC(C1(O)CC(c2ccccc2)C1)=O C1(O)(CC(=O)NC(CNC(c2c(OC)cncc2)=O)(C)C)CCCN(C)C1 c1(N2CCC(CCO)CC2)nc(N2CCC(c3ccccc3)C2)nc2c1CCC2 C1(C)(CC)COCCC1NC(=O)Nc1cnccc1Cl Cc1[nH]nc2cc(C(=O)NCC(c3ccccc3)CNC(=O)C(C)O)ccc12 C(=O)(C1c2c[nH]nc2CN1C(C1CCC(=O)C1)=O)N(CCC(O)CO)C CCCN=C(NCC(F)(F)C(C)(C)C)N1CCc2c(C(F)(F)F)cccc2C1 Cn1nc(I)cc1C(=O)NC1CN(C(c2c[nH]nc2C(F)F)=O)C1 C1(CC(N2CCC(O)(CC3(C(=O)NC4CC4)CCC3)C2)=O)CCCC(F)(F)C1 O=C(N=c1[nH]oc2cccnc12)C1CC2(CC2)CN1C(c1ccc(O)cc1O)=O CCCC(C(=O)NC(CO)C(=O)NC(C)CCC)OC C1(C(N2CCCC(OC)C2)=O)CC2OCCC2N(C(c2cncnc2C)=O)C1 CC(C)C(CNC(c1c[nH]c(=N)o1)=O)C(=O)NC(c1ccccc1)CF C(=O)(C(C)S(C)(=O)=O)N1C2CC(NC(c3cc(OC)n(C)n3)=O)(C2)C1 C(=O)(C(COC)NC(c1c[nH]c(C)c1)=O)NC1(C(=O)OCC)CC1 C1(C(=O)NC(CCCCC)C)CC(O)CCN1C(=O)CCC1CCC1 CC(C)CC(C)C(=O)NCC1CC(O)CN1C(c1cc[nH]n1)=O N1(C(c2cn(C(C)C)nc2)=O)CCC(=CCNC(C2(C)CCC(C)C2)=O)CC1 C(=O)(C1CNC(=O)c2ccccc21)N1CCC(CC=C)(NC(=O)C=CBr)C1 Cn1cc(C(=O)NC2C=CCN(C(c3n[nH]cc3C3CCC3)=O)C2)n(C)c1=O C1(CC(=O)NC2CC(CNC(=O)CC3OCCO3)C2)CCCSC1 N1(C(c2c(COC)scc2)=O)CCC(CCOC)(NC(c2cc(C)[nH]n2)=O)C1 C12(C)CCCN(C1)C(=O)CS2.C1(n2cc(C3C(COC)C3)nn2)CCCC(C)C1 c1(C(c2nnnn2-c2ccccc2)NC(C=C)(C)CC)cccc(Cl)c1OCC C1(C(=O)NCC(CNC(c2cncc(O)c2)=O)OC)CCC2(CCC2)OC1 C1(C(=O)NC2C3(NC(C=NOC)=O)CCC(C2)C3)CC(F)(F)CCC1(C)C C(=O)(C(CCOCC)NC(c1nccn1CC#C)=O)NC(CC#C)CO C=CC(CCC)CC(=O)NCC(N1CCN(C(=O)C2=CCCOC2)CC1)C(F)F N1(C(CCC#C)=O)CCC2CCN(C(c3nc(-c4cccs4)oc3C)=O)CC2C1 C1(CS(=O)(=O)NCC(C)C)CCCN(N2CCOCC2c2cccs2)C1 CC1(C)CCC=C1C(=O)NCC(O)CNC(C1CC2CCC1CC2)=O N1(C(CNC)=O)CCN(C(=O)CC2CC3(CCC3)C2)CC1.N1(C=O)CCOCC1 Cn1nnc2ccc(C(=O)NC3CC(C)(C)CCC3C(=O)O)cc12 C=C1CC(C)(C(=O)NCC=CCC(=O)Nc2cnn(CC)c2)C1 Cn1nnc2cc(-c3nc(C4CC=CCC4)nn3CC(C)(C)CO)cnc12 c1(OC)ccc(C(=O)NC2CCC(C)N(C(c3n[nH]cc3C(C)C)=O)C2)c(C)c1 C(c1cccc(F)c1)=CC(=O)N(CC(C)N(C(=O)CC1CCCS1)C)C c1(C(=O)NCCN(C(C2(CC)CCCC2O)=O)CC)cc(=O)n(C)o1 C1(NC(c2cnc(SC)s2)=O)CC2CC1N(C(=O)Cc1cocc1C)C2 CCCC(C)CC(=O)N1CCCCC(NC(c2ccc(C(=O)OC)c(C)c2)=O)C1 C1(CNC(c2c(CSCC)cccc2)=O)N(C(=O)C(C)C#N)CCC1(C)C C1(NC(c2n(C)c(S)nc2)=O)CN(C(C2CC3(C2)CC(C)(C)C3)=O)C2CCCC12 C1(NC(c2c(CC)c[nH]c2)=O)CN(C(=O)C(F)(F)c2ncccn2)CC1C c1(COCC(=O)NC(CNC(C(C=C)C)=O)C2CCC2)ccc(C)cc1 N1(C(CCCCCN(C(C2CN(C)C2)=O)C)=O)CCC(C2CCOC2)C1 N1(C(c2ccc(CC)o2)=O)CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)CC1CC C1(C(N2C(CCNC(c3ccncc3)=O)CSCC2)=O)CCC(C2CC2)C1 C1(CNC(C)Cc2cc(C3(C)CC3)on2)CCCCN1 C1(O)(CNC(COCCN(C)C)=O)CC(NC(c2coc(C(F)F)c2)=O)C1 c1(N2C3CC(CC(NC(=O)Cc4c(O)ncnc4O)C3)C2)nc2cc(Br)ccc2o1 CCC(C(=O)NCC(CCOC)NC(C1C=CCS1)=O)n1nccc1C C1(C(C)NC(=O)C(O)CC2CC2)CCN(C(=O)C(c2cccn2C)=O)CC1 N1(CC(=O)OC)C2CCC1CN(C(C(=O)Nc1ccc(F)cc1C)C(C)(C)C)C2 C#CCC(C)(C(=O)N(CCO)OC)NC(C1CC=CCO1)=O C1(NC(C(C)=C2CCCC2)=O)CCC2CN(C(=O)C(C)CC3CCC3)CC2C1 CC1C(NC(C2(CCF)CC2)=O)CCCN1C(c1ocnc1C(F)(F)F)=O N1(C(CCC2CC(NC(c3cc(C(C)=O)on3)=O)C2)=O)CCOCC1C c1(OCC(N2CC(c3ocnc3C(=O)NC3CC3C3CC3)C2)=O)ccccc1F c1(C(N2CC(CCCCNC(=O)C(O)c3ccsc3)C2)=O)cncc(F)c1Cl c1(C(N(C2C(C)CCN(C(C(C)SCC)=O)C2)C)=O)cnc2cccnc2c1 c1(OC(C)CNC(N2CCCC2c2ccc(C#N)s2)=O)ccc(Cl)cc1 CCC(CCCC(=O)NCCCSC)NC(C1CCOC1(C)C)=O N1(C(c2c(OC)ccc(F)c2)=O)CCCC2CN(c3nccc(CO)n3)CC12 Cc1ccc(C(=O)NCC(=O)NCC(CO)NC2COCC2C(N)=O)s1 C(=O)(C(O)P(C)(C)=O)N1C(CN(C(c2nc(C)nn2C)=O)C)CCC1 C=CC(CCC)CC(=O)NCCC(C)(C)CNC(=O)Cc1cc(C(F)(F)F)co1 c1(OCC(=O)NC2CCC=CO2)cccc(CNCC2CC2)c1 Cc1nn[nH]c1C(=O)NC1(CN(C(=O)CCc2nc(-c3ccoc3)no2)C)CC1 C1(CC)CCCCC1CC.C12(OCCO1)CC(=O)NCC2 C#CC1C(C(N2CCCC(NC(C3CC4(CSC4)C3)=O)C2)=O)C1(C)C C12(C(N(CCC)CCNC(C3CC3CN(C)C)=O)=O)CCCC(C1)OC2 C(=O)(CC1C(=O)Nc2ccc(F)cc21)NC(CNC(C(C(C)C)(C)C)=O)C1CC1 CCCC(C)C(C(=O)Nc1ccccc1)OC.c1(-c2cn(C)nn2)ccnc(OC)c1 C1(NC(COCc2onc(C)n2)=O)CCN(C(c2conc2C2CC2)=O)C12CC2 C(C(=O)NC(C)(CSC)C(=O)NCC1(C(C)(F)F)CC1)(C(C)C)SC c1(NC(C)C)ncc(NC(=O)Cc2cncn2C)cn1 N1(C(c2ccc(C)o2)=O)CCC(C)(C)C(CNC(c2ccccc2)=O)C1 CCCCCC(C1CC1)NC(=O)CC1(NC(=O)C=CC=CCC)CCC1 c1(C(N2C(CNC(C(C#C)(C)C)=O)C(C)CCC2)=O)onc2cc(C)ccc12 N12CC=CCC1C2.n1(C(C)(C)C)nnc(C2CC2)n1 N1(C(c2cccc(OC)c2F)=O)CCN2C(=O)C(NC(C)C)CC2C1 CC1(C)CC(NC(C2(C)CCN(C(=O)CC3CCCC3O)C2)=O)CC(O)C1 c1(OC)cc(O)ncc1C(N1CCC(C(C)NC(c2cc(O)cs2)=O)CC1)=O C(=O)(C(C)(C)CC1CCC1)N(C1CCC(NC(CC(=O)NCC#C)=O)C1)C c1(C(=O)NCC2CC(NC(C3CN(C)C(=O)N3)=O)C2)ccc2c(c1)COCO2 c1(CC)cc(C(=O)NCCCCNC(C2CCC3CC23)=O)n(C)n1 c1(C(N(CCCCCCNC(CC(CCC)C)=O)C)=O)nnn2c1CSCC2 C1(CCNC(C(C)N(C(c2coc(CO)c2)=O)C2CC2)=O)CCOC(C)C1 c1(CC(=O)NCc2snc(C(C)(C)C)n2)cccc(C2CC2)c1 c1(C(=O)NC2C(C(=O)NCCC=C)C2)c(F)cc(Br)cc1Cl c1(C(C)C)cc(CC(=O)N(C)CC2(O)CN(C(=O)COc3cccnc3)C2)on1 N1(C(CC=CC=C)=O)CCCC(CCNC(c2ccsc2OC)=O)C1 C1(C(N(CCCCC)CCO)=O)(CNC(C2(OCC)CCCC2)=O)CC12CCC2 CC1=C(C(=O)NCCC2CCCN(C(c3ccc(C)nc3O)=O)CC2)COCC1 N12CC3CCC1C1CN(CC31)C2=O.c1(C(=O)NC2CC3CCC2C3)ccnc(F)c1 n1(C(C(=O)NCCCC(C)(C)NC(C=CC)=O)C)nc([N+](=O)[O-])cc1C O(Nc1ncc(Cc2ccccc2Cl)s1)CCOC C1(NC(Cc2c(Cl)cn(C)n2)=O)COC2(C1)CN(C(c1ncn(C)n1)=O)C2 c1(C(=O)OC)cc(C#N)cnc1NCCC(C)(C)NC(c1nc(C)ncc1Cl)=O Cc1cc(=NC(=O)C(=O)NC2CN(C(C3(C)CCCCC3C)=O)CCC2C)[nH]o1 C(C(C(=O)NCC1CC2CCCC2C1)C(C)C)NC(CCC(C)=O)=O C1(CC(=O)NC2(CCC)CCOC2)CCCCN1C(=O)Cc1cncn1C C(C(O)CC(=O)NCc1cnns1)NC(CCCC1C(C)C1)=O CC1(C)CC(=O)N(CC(=O)NC2C=CCN(C(=O)Cn3cccn3)C2)C1=O C(=O)(C(CC(=O)OC)NC(=O)NC(C)C)NC1C(NC(CSCC=C)=O)CCC1 c1(OC)ncccc1C(=O)NC1CC(CNC(=O)C=CCOCc2ccccc2)C1 C#CC1CCN(C(=O)CCN(C(C2CCC3(CC3)C2)=O)CC2CC2)CC1 N1(C(=O)CCC2CCCN2C(=O)Cc2cccnc2)CCC2(CCCO2)C1 C1(NC(c2cc(CSCC)on2)=O)CCCC12CN(C(=O)CC1(CO)CC1)C2 N1(C(c2c(Cl)cn(CC)n2)=O)CCCN(C(c2ccsc2)=O)C(CO)C1 c1(CC)cnc(Cl)nc1N1CCOC(C)(CNC(c2cc(CC(C)C)c[nH]2)=O)C1 C1(C(N(CC(O)CNC(=O)CC(C2CC2)C2CC2)C)=O)CCCCC1(C)C c1(OC)cc(-c2ccc(NCc3cccc(Br)c3I)nc2)ccc1C n1(CC)cnc2[nH]c(=NCc3cnn[nH]3)[nH]c(=NC(C)COCC3CC3)c12 C1(C(=O)NC2(C#C)CC2)CCN(C(=O)CSC2CCCC2)C1(C)C N1(C(CSCC)=O)CCCC2(CNC(=O)COc3c(C)occc3=O)CC2C1.O N1(C(C2(CCC)CCC2)=O)CCC(c2n[nH]cc2CNC(C2CC=CCC2)=O)C1 C(=O)(C1=CCC(C)CC1)NC(CCOC)CNC(=O)Cc1ccc(F)cc1 Cc1cc(NC(C2C3CN(C(=O)Cn4cccc4)CC23)=O)c(O)c(C)c1 C(=O)(CC(O)CC(C)C)NC(C(=O)N(CC(CC)OC)C)C CC(O)(CC(=O)Nc1ccc(C(N2CCCNC(=O)C2)=O)nc1)CC(=O)O C#CCC(CC(=O)NCC1OC(=O)NC1(C)C)NC(=O)C=CCN(C)CC N1(C(CC=CCC)=O)CCCC1CC1CC1.C12(CCCO1)C(=O)N2 N1(C(C(COC)OC)=O)CCCCC1CNC(C1(CSC)CC1)=O c1(C(=O)NCCNC(c2nn(C)c(C3CC3)c2)=O)cc2c(F)c(F)ccc2[nH]1 C1(NC(COC)=O)CCCOC12CCN(C(=O)C(C(C)C)n1cnnn1)CC2 c1(C(N2CC3C(CNC(C(CCSC)O)=O)C3C2)=O)cnc2c(c1)CCOC2 c1(C(N2C(CNC(=O)C=Cc3cn[nH]c3)CCCCC2)=O)ccc2c(n1)NCC2 C1(COC)CN(C(=O)Nc2cc(C)n(C)n2)CCN1S(=O)(=O)C(F)(F)F c1(C(N(CC(=O)OC)CC)=O)cnc2n1CC(C(F)(F)F)CC2 Cc1cccc(-c2noc(C(C)OCC(=O)Nc3ccc(CC(C)C)nc3)n2)c1 C(C(F)(C(=O)NC12CCCCC1C2)C(C)C)NC(CSC(C)C)=O CC1(C)CCCC1C(=O)NCC1CCN1C(c1ccc(CSC(F)F)s1)=O CC1CC2CCN1C(=O)C1(CC1)CO2.c1(OCc2ccccc2)cncc(F)c1 C(=O)(CC1CCc2ccc(O)cc21)NCCOCCNC(=O)CCCF C(=O)(C#CC1CC1)NCC1(C(N(C(CC(=O)OC)C)C)=O)CCCO1 C(C(=O)N(C)CC1(C#N)CCC1)(C(C)O)NC(CCC=C(C)C)=O N1(C(c2ccc(F)cc2)C(=O)NCC(=C)C)CCC2CCC(C(=O)OC)CC12 N1(C(C=CCC)=O)CC(O)(C2CCN(C(c3sccc3SC(F)F)=O)CC2)C1 N1(C(c2ccc(F)cc2)=O)CCCC2C1CCCN2C(C1CC(C(F)F)C1)=O c1(NC)cccc(C(N2CC(C)(C)C2C2CCN(C(=O)C=CCOC)CC2)=O)n1 N1(C(c2cnc(COC)s2)=O)CCN(C(=O)C(C)(C)N2CCCCC2)CC12CC2 c1(N2CCN(C(C)=O)CC2)nc2c(c(=NCCc3nccc(C)n3)[nH]1)COC2 O=S(=O)(c1ccc(NCCOCCO)cc1Cl)NC1CCC2CCC12 N1(CC)CCC(NC(=O)C(C)(CSC)NC(c2cc(O)nn2C)=O)C1=O CC1CN(C(=O)COC2CCCCC2)CC1NC(C1CCCC1(C)C)=O C1(C(C)C)CCN(C(C2CC(CNC(=O)C(C3(O)CCCC3)F)C2)=O)CC1 C(c1nc2ccccc2o1)=CC(=O)N(CCN(C(C1(O)CCC(CC)C1)=O)C)C C1(C(Cn2cc(CONC(Cc3c(C)n(C)cn3)=O)nn2)=O)CN2CCC1CC2 C1(C(=O)NC2(CCNC(CCc3cc(C)no3)=O)CC2)CCC2CCC1O2 N1(C(C23CC(C)C2C3)=O)CC2CCCC(NC(=O)CCC34CCC(CC3)C4)C2C1 N1(C(C(C)SCCCC)=O)CC2(C1)CN(C(=O)C(c1ccccc1F)(F)F)C2 C1(CNC(=O)CC2CCCC2)CCC2(CO1)CC(NC(C1C3CCC1CC3)=O)C2 c1(NC(CN(C(C2(CN(C)C)CC2)=O)C)=O)ncc2ccccc2n1 c1(OC)ccc([N+](=O)[O-])cc1C(N1CC(C(N)=O)(CNC(C2CC2F)=O)C1)=O c1(C(C(=O)OC(c2cccc(C(F)(F)F)c2)C)O)ccc(F)c(Cl)c1 c1(C(=O)NC(C(=O)NC2C(C=C)COC2)CO)cc2ccccc2o1 c1(C(=O)NCC2C(C)C2C)ncc(N)cc1Cl O=C(CCCNCc1ccc(Cl)cc1)N=c1cc[nH]cc1F N1(C(C(c2ccnn2C)NC(c2ccnc(C)c2N)=O)=O)CCCC2OCCC2C1 N1(C(c2ccc(CNC(CCn3ncc(C)c3)=O)nc2)=O)CC2CCC(C1)O2 C1(NC(c2ncc(C)cn2)=O)CS(=O)(=O)CC1NC(c1ccc(F)cc1C)=O c1(C(=O)NCCN(C(C2CCC(C)C2)=O)C)ncccc1NCC(F)(F)F.C(C)=O N1(c2nc(OC)c(C)cn2)CCC2C1CCCN2C(c1cccc(SC)c1)=O CC(C)CC(O)CN=c1ccc(Br)c(S(=O)(=O)NCC(C)N(C)C2CC2)[nH]1 c1(CNC2CC(NC(c3ccc(CC(C)C)cc3)=O)C2)cc(F)cc(F)c1F C(=O)(C(C)CC(F)(F)F)NC1C(NC(CCC(=O)N(CCC)CCC)=O)CCC1 c1(C(=O)NC(C)CNC(=O)CN2CCS(=O)(=O)CC2)cc2c(s1)CN(C)CC2 c1(CC(=O)NCCC2(OC)CN(C(c3cc(F)c[nH]3)=O)C2)nc(F)c(F)cc1F C(=O)(C#CCNC(=O)C=C1CCCCC1)N(CCCC)C(C)CC c1(N2CC3C(C)C3C2)ccc(S(=O)(=O)NC2CCCc3ccccc3C2)c(Cl)c1 Cc1ccc(C(=O)NC2CCCC2NC(C2(C(F)F)CC(F)(F)C2)=O)cc1Cl C(=O)(CCC(CC)NC(=O)C(C)NC(=O)OC)N1CCCC(CC=C)C1 c1(C(=O)NCCN(C(=O)CC2CC(O)C23CCC3)C)cnn(C)c1S(C)(=O)=O N1(C(c2ccc(OC)cn2)=O)CCN(C(c2ccnc(CO)c2)=O)C2CCCC12 N1(C(CC2N(C(C=C(CCC)CCC)=O)CCOC2)=O)CCOC2C(O)CC12 N1(C(C(C)(C)SC)=O)CCC2(CO)CN(C(=O)Cn3nc(O)ccc3=O)CC2C1 N1(C(C(C(=O)OC)OC)=O)CCN(C(=O)Cn2cnnn2)CC1CC(F)(F)F C(=O)(C(CNC(=O)Cc1c(C)n[nH]c1C)C(C)C)NC(CCOC)C(N)=O CC(O)(CC(F)F)C(=O)NCCC1CCN(C(=O)CC(F)(F)F)CC1 C1(NC(C(CO)NC(C(C)C)=O)=O)CC2CC1CN(C(=O)C1=C(C)OCCS1)C2 N1(C(=O)Nc2ccc(OC)nc2)CCC(OC)C(C)C1.C1=COC1OC c1(C(N2CC3CC3(CNCc3c(Cl)ccc(O)c3Cl)C2)=O)cc(Cl)c(Cl)nc1Cl CC1CC2(CC(C(=O)Nc3ccnc(OC(c4ccccc4)C)c3)C2)C1 c1(CCC(=O)NCC2C3CN(C(CC4ON=C(C)C4)=O)CC32)c(F)cccc1F N1(C(CC(CCC)(C)O)=O)CCCC(C2CN(C(=O)C(C)CN(C)C)C2)C1 N1(C(CC(C)F)=O)CC(CNC(=O)COc2ccsn2)OC2COCC12 N1(C(CCC(=O)NCC)=O)CC2CC(C1)C2NC(c1cc(C)cnc1N)=O c1(C(=O)NCC2C(C)CN(C(c3ccoc3Cl)=O)CC2)cnn2c(N)ccnc12 N1(C(CC(C)SC)=O)CCC(=CCNC(=O)CCc2cnoc2)CC1 C(CC(=O)NC1CC(NC(=O)C(C)(C)C2CCCCO2)C1)(c1cccs1)N(C)C C1(NC(c2cccc(CC)n2)=O)CN(C(c2cc(C(F)F)no2)=O)C(C)(C)C1 CCC(CC)CCCC(=O)N1CCCC1CC(=O)NCC(C)C1CC1 c1(C(=O)NC2C(CNC(CC=C=C)=O)C2)cccc2c1NC(=O)CO2 N1(CCNC(C(C2CCCO2)NC(C=CCOC)=O)=O)CCOC1=O c1(C(=O)NC(CCCNC(c2cccc(OCC)c2)=O)C)ccc2ccnn2c1 c1(CC(C(=O)OCC)NCc2ccc(O)c(O)c2)ccc(O)c(I)c1 C(=O)(CCC(F)F)N(C)CC1CN(C(C(C)SCC2CCCO2)=O)C1 C1(CC(=O)NCC(N(C)C(c2cnc3n2CCS3)=O)C2CC2)CCC(C)(C)CC1 c1(C(=O)NCC2CC(C)N(C(=O)CC(=O)N(C)C)C2)ccnc(Cl)c1N c1(OCC(N2CC(c3cn(CCCCO)nn3)C(O)C2)=O)ccc(F)cn1 C1(NC(=O)CCn2ccnn2)CC2CC1CN(C(c1cncc3ccsc13)=O)C2 c1(C(=O)NCCCC(CO)NC(C(COC)N(C)C)=O)cc(Cl)c(C)cn1 c1(NC(=O)Nc2c(C)nc(CCC)s2)c(C)cccc1Cl C(C(=O)NCC(C)CN(C)C(c1cscn1)=O)(C1CCCC1)OC Cc1nc2cc(C(N3CCC(NC(c4ccccc4)=O)C34CC4)=O)c(F)cc2[nH]1 O=C(C1COc2ccccc21)N1CC2CC(C1)C2NC(C1(CCF)CCC1)=O N1(OCCOC(=O)NC2CC2NC(c2cccc(CO)c2)=O)CCCCCCC1 C1(CCCNC(c2nsnc2O)=O)CCCN1Cc1nc(-c2cccnc2)no1 C1(NC(C(n2cc(Cl)cn2)C)=O)CC2CC1CN(C(c1cnsc1)=O)C2 N1(C(CCC2(C)CC2(F)F)=O)CCCC(F)(CNC(=O)C2=NOCC2)CC1 C1CCCCCCC(=O)N1.Cc1cccc(-c2cn(C(C)C(=O)O)nn2)c1F CC(C)C(C)(CNC(C1CC=CCC1)=O)NC(=O)CCc1cncnc1 n1(CCc2c(CC)cccc2)cnc2c(N3CCOCC3CCO)ncnc12 C1(CC)(NC(C2CC(SC)C2)=O)CCCN(C(=O)C(C)Oc2ccccc2F)C1 CN1CCC(C(N2CCC(CCNC(c3nocc3Cl)=O)CC2)=O)CC1=O c1(OC)cccc(OCCOC(C2CC(C(=O)O)C2)=O)c1 N#Cc1cncc(C(N2CCC(C(=O)NOCCc3ccccc3)(CF)C2)=O)c1 C1(CNC(CCSCC(N)=O)=O)CN(C(c2csc3nccn23)=O)CCCO1 C1(C(F)(F)F)(C(N2CCN(C(COCCC#C)=O)C(C)C2)=O)CC2C=CC1CC2 C1(C(N2CC(O)(CNC(C(C)=CC)=O)C2)=O)CC2CCC1CC2 Cn1cc(C#CCNC(=O)NCc2ccc(Cc3ccc(F)cc3F)cc2)cn1 CCC(CC(=O)NCC1(O)CN(C(C2CC(F)(F)CCC2(C)C)=O)C1)C(C)(C)C N1(Cc2cc(C)ncc2)CCC2(CC1)CC(C(=O)NC1CCCCC1)C2 c1(C(N2C3CN(Cc4c(C)cc(Br)cc4C)C(C3)C2)=O)c(Cl)ccc2c1OCO2 C12(C(N3CCC(C(C)NC(=O)CC4CC5CC5C4)C3)=O)CC3CC1C2C3 C=CCC(C)C(=O)NCCC1(CNC(=O)CCSCc2csc(C)n2)CC1 c1(C(=O)NC(CC=C)CNC(C2(C)CC=CCC2)=O)cnc(O)c(Cl)c1 C(C1=NOC2CN(C(=O)COCCN(C)C)CC12)NC(C1CCC(F)(F)CC1)=O c1(C(N2CC(N(C(=O)Cc3ccco3)C)C2)=O)scnc1C1CC1 C1(NC(c2cc(OC)ncc2)=O)CC(O)CN(C(c2cc(C)nc(O)c2)=O)C1 C=CC(C)(O)CC(=O)N1CC(C(F)Cn2cc(-c3cncs3)nn2)C1 CC1CCCC(O)(C(N2CC(CCNC(C3(F)C(C)(C)C3(C)C)=O)C2)=O)CC1 C(=O)(C(F)(F)CO)NN1CCCC1NC(=O)OC(C)(C)C.C1(C(C)N)(CC)CC(=C(C)C)C1 c1(CC)cncc(C(=O)NC(C)C(=O)NC(C2CCC(NCS(C)(=O)=O)C2)=O)c1 n1(CC(=O)NCCCC(C)NC(=O)C(C)c2cccs2)ccc2cccnc12 Cc1ncc(C(=O)NC2(CNC(=O)C(O)CNC(=O)OC(C)(C)C)CCCC2)o1 C1(NC(=O)CN2CCCS2(=O)=O)CCCCCN(C(C2CC3CC3C2)=O)C1 C1(C(C)NC(c2c[nH]c(Br)c2)=O)CCCN(C(c2cscn2)=O)C1 c1(C(=O)NCC2(C)CCN(C(=O)CO)C2)ccc(Br)c2cn[nH]c12 N1(C(c2cc(OC)ncc2)=O)CCN(C(=O)Cc2ccoc2)C(C)CC1C c1(C(N2C(CCNC(CCOC)=O)CCCC2)=O)ccc(OC(C)C)c(Cl)c1 N1(C(CCOCCOCC)=O)CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)C(C)C1C c1(-c2cccc(NC(=O)CC3CCCCO3)n2)cccc2ccoc12 N1(C(CC=CCC)=O)CCCC(NC(=O)CC(O)c2ccccc2)C1 C1(NC(=O)CN2CC=CC2)C2CC1N(C(=O)C(O)Cc1cc(Cl)sc1Cl)C2 c1(C(=O)NCC2(CO)CCN(C(CCC(C)C)=O)C2)ccc(F)c(N)c1 C1(C(=O)NC2CC(NC(Cn3c(C)ccn3)=O)C2)CN(C)CCO1 C1(C2=CCCCCC2)(C(=O)NCC2(C)CN(C(C=COCC)=O)C(C)(C)C2)CC1 c1(C(=O)NCC2CCC(C)N(C(c3cnc(Cl)cn3)=O)C2)cc(N)c(N)cc1F c1(-n2cc(C3(NC(c4cc(C)c(C)o4)=O)CCC3)nn2)cccc2sccc12 c1(OC)ccc(C(C)CNC(C2(C(=O)O)CCCO2)=O)c(C)c1 C1(CCNC(C(CC)OC2CCCC2)=O)C2CN(C(=O)C(Cl)=CCl)CC12 c1(C(=O)NC(C(C)NC(c2cc[nH]c2C2CC2)=O)C)cc2c(F)ccc(F)c2[nH]1 c1(C(=O)NC2(C)CN(C(c3ncn4c3CCC4)=O)C2)nccn2cnnc12 N1(C(c2cc(OCC)n[nH]2)=O)CCC(NC(=O)C2=CCSC2)C1(C)C c1(C(=O)NC2CCCC(NC(c3cc([N+](=O)[O-])c[nH]3)=O)C2)n[nH]c2c1CCOC2 C1(C(=O)NC(C(=O)NCC)C)CN(C(=O)C2=C(Cl)CC2)CC1CC C(=O)(C1=C(CCl)N(c2ccc(Br)cn2)C(=S)NC1c1cc(C)nn1C)OC Cc1sc(=NCc2cn(-c3c(F)ccc(Br)c3F)nn2)[nH]c1C1CC1 N1(C(C(C)=O)=O)CCCN(C(=O)COCc2cccc(C)c2)CCC1 C1(NC(c2c(OC)csc2)=O)CCC2CCN(C(C3(C)CCN(C)CC3)=O)C12 CCC(C)CC(C(=O)NCc1nnnn1CC)NC(C1CC(=C2CC2)C1)=O c1(C(N2CC=CC(NC(C3C(C=C)CC3)=O)C2)=O)ccc(C)c(CO)c1 c1(SC)c(O)cccc1F.C12C(CC)CCN1C(=O)CN(C(C)(C)C(F)(F)F)C2=O N1(C(c2cc(C)c(N)cn2)=O)Cc2[nH]nc(C(=O)NC3CCCSC3)c2C1 c1(C(=O)NC(CC=C)CNC(c2ccnc(OC)c2)=O)ncc(Cl)cc1Cl c1(C(N(CC(C)NC(=O)Cc2ncc(C(F)(F)F)[nH]2)CC)=O)cn2ccnc2s1 N(C1CCOCc2c(Br)cncc21)C(N1CC(=O)N(CC2CCCC2)CC1)=O O=C(C1c2ccccc2CN1Cc1ccnc(Br)c1)Nc1ccc(CCl)nc1 C1(C(=O)NC2(C#N)CCN(Cc3c(OC)cccc3C)C2)Cc2ccccc2O1 C1(OC)CCCC(CC(=O)NCC=C2CCN(C(=O)CCC=CBr)CC2)C1 C=CC1(C(=O)NCCN2CCOCC2C)CCN(C(=O)CCC(C)(C)OC)C1 C(=O)(C(C)CCC(C)(C)C)NC(CCOCC)C(=O)NC(CC)C1CCC1 C(CN=c1nc(N2CCC(C)(C)C(CO)C2)c2c([nH]1)CCOC2)=CCCC Cc1cc(Br)cc(F)c1C(N1CCC1(C)C(=O)Nc1ccnc2c1CCO2)=O c1(C(C)SCC)nc(-c2cc(CC)c(C)s2)n(CC2CC(C)C2)n1 C1(CNC(C=C(C)C)=O)CCCCCN1C(=O)C(C)n1ccnn1 C12(C(=O)NC(C)CCCNC(=O)CCCCC(N)=O)CCCC(=O)N1CCC2 C1(CC)C(NC(=O)C(O)CCCN(C)C)CCCN1C(=O)CSc1nncs1 N1(C(C2CC(SC)C2)=O)CCN(C(c2cnn(C)c2)=O)C2CS(=O)(=O)CC12 N1(C(CCCOCC=C)=O)CC2CCC1C1CN(C(=O)C(C(C)C)N(C)C)CC21 N1(C(c2cc(C)ns2)=O)C2CCC1CC(NC(c1ccc(OCCF)cn1)=O)C2 C=CCN=c1nc(N2CCOCC2)[nH]c(=NC(C)c2cnns2)[nH]1 N1(C(CC2(OC)CCC2)=O)Cc2ccccc2C1C(=O)Nc1cccc(Cl)c1F N1(C(c2n(CC)ccn2)=O)CC(NC(=O)CC2CC(F)C2)C2CCCCC12 CCCN=c1cc(C)c(S(=O)(=O)NC2(c3cccnc3)CC3(CCC3)C2)c[nH]1 c1(C(=O)NCC(C(C)C)(C)NC(=O)CC2CCSCC2)ccccc1S(C)=O c1(C(N2CC3C(NC(CC=C=C)=O)(CC3)C2)=O)ccc(C)c2ccccc12 C1(C(=O)NCCCCOC(=O)C(O)C(F)F)CCCN(CCNCCCNC)C1 C1(CNC(CCCC#C)=O)CC(C)CN(C(c2coc(CC3CC3)n2)=O)C1 c1(C(N2CCN(C3CN(C(CC(COC)C)=O)C3)CC2)=O)cnn2c1CCCC2 N1(C(CC2N(C(c3cc(C)c(F)cn3)=O)CC2)=O)CC2(CC(CO)CO2)C1 C12(NC(CCNC(COC)=O)=O)CCCC1N(C(=O)CC1C(C)(C)C1(C)C)CC2 C=CC1CC(NC(C2(NC(=O)CC(=O)OCC)CC2(C)C)=O)C1 C1(NC(Cc2c(C)cco2)=O)CCN(C(c2coc(C3CC3)n2)=O)CC1O O(N1CCC(CC(=O)NC(CNC(C2CC(F)C2)=O)CC(F)(F)F)CC1)CC c1(C(=O)NC2(CNC(C3(C(F)F)CC3)=O)CCCCC2)cc2c([nH]1)CCCC2=O c1(SC)ccc(C(=O)NC(C)CNC(c2ccc(=N)[nH]c2)=O)cc1Br C1(C(=O)NC2CC=CC2)CCN(C(=O)C2=C(Cl)CCOC2)C12CCC2 c1(C(=O)NC(CCOC)CNC(C2CCC(CSC)C2)=O)cccc(N)c1F C1(N=[N+]=[N-])(C(=O)NC2C(C)COCC2)CCN(C(C2CC(O)CN2C)=O)C1 N1(C(C)=O)CCC(c2cn(C3(C(=O)Nc4cc(=O)n(C)cn4)CC3)nn2)C12CC2 C1(NC(COCc2c(C)cccc2)=O)CN(C(c2ccnnc2S)=O)CCC1C C1(C(=O)NCC(C)(C2CC2)NC(=O)CC2(N3CCCC3)CC2)CC(=O)C12CCCC2 C1(C(=O)NCC2CCC(C(N(C3CCCC3)CCC)=O)CC2)CCCC2(CC2)C1 C(=O)(C(C)C(C)(C)C)NC1(C(=O)NCC(COC)(C)O)CCOCC1 C(c1ccc(C(N)=O)o1)=CC(=O)NC1C(CN(C(=O)Cn2nnc(=N)[nH]2)C)C1 O(N1C(=O)c2ccccc2C1=O)CCNC(N(C1COCC1(C)C)C)=O N1(C(c2cnc(CCC)s2)=O)CCC(C)C(CNC(c2nn(C)cc2Cl)=O)C1 C1(C2CCC2)(C(N2CCC(F)(CNC(CC(CC)SC)=O)CC2)=O)CC1(F)F C=C1Cn2c(Cc3nc(CCO)nn3-c3cccc(Br)c3)nnc2S1 C=CC(C)CC(=O)N(C)CCN(C(=O)C(C(C)C)Sc1ccccc1)C CCCCC(C)(F)C(=O)NCC(O)CC(=O)NC1C=CC(C(=O)NC)C1 Cc1cnc2cc(C(N3CC4CC4(NC(=O)CCc4cc(Cl)cs4)C3)=O)ccn12 N1(C(C=CC(=O)N(C)C)=O)CC2CCC2(CC(=O)N(C2CCCCC2)CC2CC2)C1 CC(C)(CC1CC1)C(=O)N1CCC(CNC(C2CC3CCC2C3)=O)C1 CC1CC(C(=O)NC(CCN(C)C)C(=O)N(C)CC2CCCS2)CN1C C(C(C)(C)CNC(=O)C(F)OC(F)(F)F)N(C(=O)CCCc1n[nH]c(=N)s1)CC C(=O)(C(C)C(C)O)N1CC(NC(C(C)C2CCCC2)=O)(CO)C1 C1(CN(C(C(=O)NCC)=O)CC)CCN(C(c2ccon2)=O)CC1 c1(C(=O)NCCOC2CN(C(C(c3ccnn3C)C)=O)C2)ncc(F)cc1N C1(C(=O)NC2(C)CC(NC(C3N(CC)CCC3)=O)C2)Cc2ccc(F)cc2C1 Cc1cc(C(=O)NCCCCC2(NC(=O)C(N)=O)CC2)n(C(C)(C)C)n1 Cc1nccn1C(C)C(=O)NC1CC(CCNC(C2CC(O)C2)=O)C1 c1(C(=O)NCC2(NC(=O)CCCCN3CCCCC3)CC2)ccc([N+](=O)[O-])cn1 c1(C(N2CC(C(N3CCC(n4cccn4)C3)=O)C(F)C2)=O)nccc2[nH]ccc12 N1(C(C)=O)CCOC(C(N2CCCC(NC(C3(C#N)CCCC3)=O)C2)=O)C1 c1(CC(=O)OCC(C2CC2)OCC)cncc2ccccc12 C1(c2cn(-c3c(CC)scc3)nn2)CC(C)CCN1C(=O)C(C)CC C(=O)(CCCC(CCC)CCC)N1CCCC(NC(CCCCCC#C)=O)CC1 C(CCCCCC(=O)NC(C)(C)C(C)NC(=O)C=Cc1cccnc1)SC N1(C(C)=O)CCC(c2ccc(OC)cc2)C(NC(=O)Cc2ccc(O)c(C)c2)C1 C(=O)(CC(C)C(F)(F)C(F)(F)F)NCCN(c1cc(SC)ncn1)CC C1(C(=O)NCCN(CC=C)CC)C=CCOC1 C(=O)(C(F)C(C)(F)F)NCc1cn(C2CN(C(COC(CC)C)=O)C2)nn1 C(=O)(C1=CCCOC1)N1CC(O)(CCNC(=O)C(c2ccc(Cl)s2)=O)C1 O=S(=O)(C1CC12CCC2)NCc1nc(COc2ccccc2)cs1 C12(CNC(C3N(C)C(=O)CCC3)=O)CCCC1CN(C(C1CC(C3CC3)C1)=O)C2 c1(C(=O)NC(C(CC)C)C(=O)NCCc2nncn2C)ccn2ccccc12 c1(C(=O)NCC(CNC(c2cc(C)nc(C)c2)=O)(C)O)ccc2cc(C)cn2c1 N1(C(c2c(C(C)C)onc2)=O)CCCC(C2CN(C(c3cncc(Cl)c3)=O)C2)C1 c1(C(N2CCN(C3CN(C(CNC(CC)=O)=O)C3)CC2)=O)ccnc(F)c1Cl C=CCC(C(=O)NC1CCC(C)N(C(c2ncccc2F)=O)C1)C(C)C N1(C(=O)COCc2cccnc2)C(CNC(c2cc(Br)c[nH]2)=O)CC2COCC12 c1(C(N2CCCC(C)(NC(C3C(C)=C3)=O)C2)=O)ncc([N+](=O)[O-])n1C N1(C(C23C4C5C(C(=O)NCCOC(F)(F)F)C(C2C4)C53)=O)CC2CCCC(C2)C1 CC(C)CC(C)CC(C)C(=O)NCCCNC(c1cn(C)nc1C(F)F)=O c1(C(N(C(CN(C(C(CC)(C)C)=O)C)C)C)=O)cc(O)nc(C)n1 C(=O)(CS(N)(=O)=O)NC1C(NC(C(=O)NC(C)C)=O)CC1 C1(NC(C(Cc2ccco2)NC(c2cc(C)[nH]n2)=O)=O)CN(C)CC12CC2 C1(S(=O)(=O)c2ccccc2)(C(N2C(Cc3cn(C(C)C)nn3)CCC2)=O)CC1 c1(CC)cc(C(=O)NCC2CCC2NC(C2CCCOCC2)=O)oc1CC N1(C(c2c(C)n(C)cc2)=O)CC(C)(C)CC1CNC(C1CCC(CN(C)C)O1)=O C1(C(N(C(C)CCNC(=O)C(F)=CC2CC2)C)=O)CC12CCCCCC2 N1(c2nnc(CC)o2)CC2(CCCC2NC(c2cc(O)nn2C)=O)C1 N1(C(C(C)n2cccn2)=O)CCC(O)CC1C(=O)NCC1(F)COC1 CCCC(C)C(=O)NCCOC1CCN(C(c2cnc(CCC(F)(F)F)s2)=O)C1 c1(C(N2CC(OC)C(NC(C34CC(C)C3C4)=O)C2)=O)cccc(C(F)F)c1F C1(CCC)CN(C(=O)CSc2nncn2C)CCN1C(=O)CP(C)(C)=O N1(C(C(=O)Nc2ccc(C(=O)OC)c(Cl)c2)=O)CC2COC(C)(C)OCC2C1 C1(CN(C)C(C2(C3CCCO3)CC2)=O)CCN(C(c2ccnc(CO)c2)=O)CC1 CCC(CC)C(C(=O)NC1CC1)OCc1cnn(C)c1C(=O)N(CCCO)OC c1(C(=O)NCc2c(C(C)C)con2)cc(CNC(C2CCCS2)=O)ccn1 C1(NC(CCOCCN(C)C)=O)CC(F)CN(C(=O)CCCC2CCCC2)C1 c1(N2CCC(C)CC(C)C2)nc2cccnc2c(=NCc2cc(Br)cnc2Br)[nH]1 CC(C)(N)CC(=O)N1CCOCC1.C(C(F)F)N N1(C(CC(C=C)C)=O)CCC(NC(c2ccc(O)cc2)=O)CC1C Fc1ccc2c(c1)C(N1CCC(Nc3ccc4ccccc4c3)CC1)CC2 c1(OC)ccc(C(N2CCN(C(C3CC=CC3)=O)C(CF)C2)=O)c(O)c1 c1(CNC(CC(C(=C)C)O)=O)ccc2c(=N)[nH]oc2c1 C1(O)(CC(=O)NCC2CCN2C(=O)CCn2ccnc2)CCOC1 N1(C(C(C)(C)OC(C)=O)=O)CCN(C(=O)CN2CCN(C3CC3)C2=O)CC(O)C1 N1(C(=O)NC(c2cc(C(F)(F)F)n[nH]2)C)CCC2CCCC(C2)C1 c1(C(=O)Nc2ccc(C)cc2)nc2n(c1Cl)CCN(c1nccn1C)C2 Cc1c(C(=O)NCCC2CC(NC(=O)CCN(C)C)C2)cncc1Br CC1(C(=O)NC(CNC(=O)CC2CCCC2)C2CCC2)CCC1 N(C1CCS(=O)(=O)c2ccccc21)C(=O)Nc1ccc2c(c1)OCC(=O)N2 n1(CCOC)nnnc1C(c1sccc1Br)NCC1CCCCC1 C1(C(N2CCC(F)CC2)=O)CCC(C2CC2)N1C(c1ccccc1CO)=O c1(NCCCCOCC)cc(Br)ccc1S(=O)(=O)NCCC1CCCCC12CC2 Cc1ccc2[nH]c(=NCCN(C(C3(C)CCCCNC3=O)=O)C(C)C)sc2n1 N1(C(C2C(CC)CCC2)=O)CCCC(C)(CNC(c2occc2Br)=O)C1 C(=O)(C1=CC(C)(C)C1)NC(CC#C)C(=O)NCc1ccnn1C O=S(CCN1CCCC(CF)C1)c1ccccc1 Cc1cc(C(=O)NC(CCF)C(=O)NCC2CN3CCC2C3)oc1C c1(CC(C(=O)OC)n2nnnc2C)c[nH]c(=NC2CCCN(C)CC2)cn1 C1(CNC(C(C)OCCCC)=O)CCCN1C(c1scnc1C(C)(C)C)=O N1(CCc2cn(C(C(N3CCC(OC(C)=O)CC3)=O)C)nn2)CCS(=O)(=O)CC1 N(C1CCCSc2ccc(Br)cc21)CC(=O)OC(C1CCS(=O)(=O)C1)=O N1(C(c2cc(C(C)C)no2)=O)CCC2CN(C(=O)CCC3CC3(Cl)Cl)C2C1 c1(C(=O)NCC(CNC(C=CCC)=O)C)ccc(-n2cnnn2)cc1 C(CC(C)C)(C(C(=O)NCC(F)F)N1Cc2ccc(N(C)C)cc2C1)OC C1(NC(C2CCCN2C(c2ccc(Cl)nc2F)=O)=O)CCCCC1(F)F N1(CCc2ccc(OC)cc2Cl)CCCC2(CC1)CNC(=O)O2 N1(C(=O)COc2ccccc2CCCCCCCO)CC2CCOCC2(CO)C1 C(=O)(CCS(N)(=O)=O)N(C1CCN(C(=O)CCC(=O)NC2CCCC2)C1)C CC1=C(C(=O)NC2CCC2NC(=O)C=C2CN(C(=O)OC(C)(C)C)C2)CCO1 C1(O)(CC(=O)N(C)CC2N(C(CCc3nc(C)sc3)=O)CCC2)COC(C)(C)C1 C1(C(N2CC3CC3(CO)C2)=O)CC(c2cc(F)ccc2F)=NO1 N1(C(C2C(CC)CCC2)=O)CCCCC(CN=c2nc(-c3ccccc3)[nH]s2)C1 C1(OC)(OC)CC(C(=O)NC(C)CNC(c2cc(CN(C)C)no2)=O)C1 Cc1nc(NCC2CN(C(c3cscn3)=O)CC2C(F)(F)F)ccc1[N+](=O)[O-] c1(CC)[nH]ccc1C(=O)NCC1CCN(C(=O)COCc2nc[nH]n2)C1 C1(NC(C(C)OCC(C)C)=O)CCN(C(c2cnc(OC(C)C)s2)=O)CC1F C1(CC(N2CC(NC(c3cccs3)=O)(CF)C2)=O)CC(C2CC2)C1 c1(C(=O)OC)ncc(C(=O)NCC2CC2NC(c2ccc(NC(C)=O)s2)=O)s1 N1(C(C(=O)OCC)=O)CC(OC)CC(NC(=O)CCC=Cc2ccccc2)C1 N1(C(c2cc(F)n[nH]2)=O)CCC2(COC(CNC(C3(O)CCC3)=O)C2)C1 C1(CC(=O)N(CCCCN(C(C2(OC)CS(=O)(=O)C2)=O)C)C)OCCCC1(C)C CC1(C)C2CC(C(N3CCCC3(C)CCC(=O)NCC3(C)COC(=O)N3)=O)CC12 C(c1cnn(C)c1)=CC(=O)NC1C(CC(=O)NC2(C)CC(C)C2)C(O)C1 n1(CC#C)c(C)cc(C(N2CCN(C3CN(C(=O)C=COCC)C3)CC2)=O)c1C CC12CC(C(=O)NCCCCNC(C3CCN(C4COC4)C3)=O)C3CC1C2C3 N1(C(CCN(CCC)C(CCC(C)C)=O)=O)CCOC(CC(=O)NC)C1 C(=O)(CC(O)CCC)NCC1(NC(CCC=C)=O)CCCCC1 c1(C(=O)OC)cc(Br)c(CNC2CCN(Cc3ccncc3)C2)s1 C12(CNC(CCC(CC)OC)=O)CCCC1CN(C(=O)COC1(C)CCCC1)C2 Cc1cc(C(=O)NC2CC3(C2)CC3NC(c2cncc(Cl)c2)=O)cc(O)n1 c1(C(N2CCN3CCOCC3(COC)C2)C(=O)NCC)ccc2ccc(Cl)cc2n1 c1(NC(CCNC(C2CC(OCC)C2)=O)=O)ccc(OC)c(O)c1 C(C)(C)(CCC(=O)NCC1CC(F)CN1C(=O)CC1CNC(=O)O1)N(C)C C1(C2CCN(C(=O)C(O)c3ccsc3)CC2)(NC(C(C)(C)C(F)F)=O)CC1 N1(S(CC2(C(C)C)CCC2)(=O)=O)CCC2(CCNCC2)CC1 c1(OC)ccnc(NCC2C=CC(NC(=O)CCOCC(F)F)C2)n1 c1(C(N2CC(CNC(C(c3n(C)ncc3)(F)F)=O)C2)=O)cc(N)c(F)cn1 c1(C(C)=O)ccc(C(N2CCCCC2CCNC(=O)CC(C)C(C)C)=O)c(F)c1 N1(C(CCOC2CN(C(=O)CCc3ccc[nH]3)C2)=O)CC2(C=CCO2)C1 c1(C(=O)NC2C3(CN(C(c4cc(C)on4)=O)C3)CCC2)n[nH]c2c1CC(C)CC2 Cc1cc2cc(C(N3CCC(C)C3CNC(c3cn(C)cn3)=O)=O)oc2cc1C O=C(CCCCc1cccnc1)NNc1cccc(F)c1Br c1(C(=O)NC2CC(CNC(C(CC)(C)O)=O)C2)c(Cl)cc(Cl)cc1Br C(c1cccc(F)c1Cl)=CC(=O)NC(CNC(C1CCN(C)CC1)=O)C1CC1 CC1(C(=O)NCC(O)CF)CCCN(C(C2CCCCC2)=O)C1 c1(C(C(=O)NC2CCOC2)N(CCOC)C2CC2)ccc(OC)nc1C c1(C(=O)NCC2CC(NC(CCc3n(C)cnc3)=O)C2)cc2ccncc2s1 C1(C(N(CC(C)(C)NC(C2CCC(C)(C)O2)=O)C)=O)CCC2(CCCO2)CC1 C=C(Cl)CC(N)C(=O)N(C(c1ncccn1)C)CC c1(C(N2C(CNC(COCCOC)=O)CCCC2)=O)cncc2cnccc12 c1(C(N2CCC(NC(c3c(C)cc(O)c(Cl)c3)=O)C2)=O)cn2c(n1)C(C)CCC2 c1(-c2nc(CC3CC(OC)C3)n(C(C)C)n2)ccc(N(C)C)c(Cl)c1 c1(C(=O)NCC(CNC(c2ncn(C(C)C)c2)=O)(C)O)cccc(N(C)C)c1 c1(CC(=O)NC(C2CCCC2)CNC(C(CC)O)=O)ccc(C(=O)NC)nc1C c1(OCC)cc(Br)c(F)cc1NC(=O)NCC1CCCCC1F c1(OC)nc(=NCC2CCCN2C(=O)C=Cc2ccc(F)cc2)nc(OC)[nH]1 C1(C(=O)NC(c2ccns2)C)CCN(C(=O)COCCN(C)C)C(C)(C)C1 C1(c2n(C(CC)C)nnn2)(NCc2csc(C(C)(C)C)n2)CCCC2(CC2)C1 c1(CC(=O)NC2C(CNC(C3ON=C(C)C3)=O)CCC2)c[nH]c2ccc(C)cc12 CC(CN=C(NCC1CC(OC(F)F)C1)NC1CCC1)N1CCCCC1 c1(C(=O)NCCC(C)NC(c2cc(CC)on2)=O)c[nH]c2c(Cl)cccc2c1=O C(=O)(C(Cc1ccccc1)C(C)O)NCCn1ncc(CC)c1.C(C)(C)(C)OC(C)=O C12(NC(C=CC(=O)N(C)C)=O)CCCC1CN(C(=O)CN1OC(C)(C)CC1=O)C2 C1(C2CCN(C(=O)C(C)CN(C)C)CC2)(NC(c2c(C)cc(F)cc2)=O)CCC1 Cc1[nH]c(C)c(C(N2CCC(C(C)C(=O)NCC3(N(C)C)CCC3)CC2)=O)c1C N1(C(CC2C=NN(C)C2=O)=O)CC(NC(C2(O)CCCCC2)=O)CC(C)(C)C1 c1(OC)cc(CC(=O)N(C)CCN(C(=O)CC2CCCO2)C)cc(Cl)c1 c1(C(=O)NCCC(C)NC(CN(C(C)=O)C)=O)ncccc1N=[N+]=[N-] c1(OC)cccc2c1C(C(=O)N(CCNC(c1cncs1)=O)CCN(C)C)CC2 c1(C(N2CC(SC)C(NC(=O)C=C(C)Cl)C2)=O)ccc2c(c1)CCC2(C)C C1(CNC(N(C2CN(C(C)C)C2)C)=O)CCc2nn(C)cc2C1 n1(CC(=O)NC(CN(C(c2ncc(OC)cc2F)=O)C)C)ncc2cccnc12 C(CNC(c1[nH]ccc1C)=O)(CC(=O)NCCC1CCCCCC1)OC c1(C(=O)NC(CC(C)NC(Cc2cnc(C)[nH]2)=O)C)cccc(CC#N)c1 CC(CNC(c1nnc(S)n1C)=O)C(F)C(=O)Nc1ccc(F)c(CO)c1 c12ccc(cc1)NC(=O)N2C(C)(C)C.CCC#CCCN C1(C(=O)OCc2ccc(-n3c(=O)cc(C(=O)OC)[nH]3)nc2)CC(=O)OC1(C)C c1(NCC(=O)NC(C(=O)NCCC2CC(F)(F)C2)c2ccco2)ccccn1 C(=O)(C(Cc1ccc(N)cc1)S(C)(=O)=O)N1CCC(C2C(C)(C)CO2)CC1 C1(NC(C(CC)OC)=O)(CO)CCCN(C(=O)Cc2ccc(Cl)c(Br)c2)C1 N1(C(C2(C)C=CCC2)=O)CCC(C(O)CC(=O)OC(C)(C)C)CC1 c1(C(=O)NCC2C(C)CCN2C(=O)CCC(C)(C)C)cc2ncc(Br)cn2n1 Cc1[nH]nc2ncc(C(=O)NC(C)C(C)NC(=O)C(F)(F)C3(O)CCCC3)cc12 c1(CCC(=O)NCC(C)N(C(C=C(C)C)=O)C)cccc(F)c1 n1(CCC(C)C)cc(C(=O)NCC2CC2NC(=O)CCc2cscn2)nn1 C(=O)(CC(C(F)(F)F)NC(=O)CCCCCC#N)N(C)CC1CCN(CC)C1 Cc1cncc(C(=O)NCC(F)CNC(=O)C(c2cccc(Cl)c2)O)c1C C12(Nc3ccc(C(=O)OC)nc3OC)CCC(C(=O)OC)(CC1)CC2 c1(CN2C(COC)CN(C(=O)Cn3cc(Cl)cn3)CC2)cccc(F)c1[N+](=O)[O-] C(C(CC(=O)N1CCC(CO)C1C)NC(=O)C(C1CC1)SC)OC C=CCCN=C(NC1CCCC1(F)F)N(C)Cc1ccccc1C(C)C C1(NC(c2ccn3ccnc3c2)=O)CCC2(CC1)CN(C(C1CC1Cl)=O)CCO2 c1(C(N2CCC(NC(C3(C=C)CC3)=O)C2)=O)ccc2c(c1)SCC(=O)N2 c1(-c2c(OC)ccc(F)c2)cc2c(C(=O)Nc3ncco3)coc2cc1N c1(C(=O)OC)ccc(CC(=O)NC2CCC(NC(c3sccc3CO)=O)C2)cn1 C(=O)(C1=CC2(CCN(C(=O)CCCn3cc(CN(C)CC)nn3)CC2)OC1)OC C1(CNC(c2c(C)ccc(C)n2)=O)CCCC2(CN(C(=O)C(C)C3CCC3)C2)O1 c12ccc(cc1)-n1cc(nn1)C2.c1(CNC(=O)Cn2cc(I)cn2)ccccc1 c1(C(N2CC(CCNC(COCC#C)=O)OC(C)C2)=O)cc2cc(C)ccc2o1 N1(C(C(C)C(F)F)=O)CC(C)OC2(CCN(C(=O)CCc3cnco3)CC2)C1 c1(OC)ccnc(C(=O)NC2COCC2CNC(=O)Cc2[nH]cnc2C)c1OC N1(C(C2(O)CCCCC2)=O)CC2CCN(C(C3(O)CC4CCC3C4)=O)CCC2C1 C(=O)(C1=CCCOC1)NC(C)(C)CN(C(=O)OC(C)(C)C)Cc1cccc(I)c1 c1(C(N(C2CCN(C(=O)Cc3ccsc3C)C2)CC)=O)cn(C)ccc1=O N1(C(Cc2n(C)nnc2)=O)CCCC2(CCCCC2NC(=O)C=C(Cl)Cl)C1 C1(COC)CN(C(c2ccncc2Cl)=O)CCN1C(=O)CC(F)(F)Br N1(C(CCOCC)=O)CCN(C(=O)CNC(C2CC2C)=O)C2(CCC2)C1 N1(C(C2(CC)CCCN(C(C3CCS3(=O)=O)=O)C2)=O)CCC(CO)C(C)(C)C1 C1(CC)C(NC(c2ccc(N)cn2)=O)CCCN1C(=O)CCC1CCOCC1 CC1CCC(C(N2CC(OCCNC(c3csnc3Cl)=O)C2)=O)C1 C1(NC(C(CC)NC(C)=O)=O)CC2(C1)CC2C(=O)NC(c1cccs1)C C(C)(CO)(C(=O)NC(C)CCNC(c1ccc(N)cn1)=O)OC Cc1cc(C(=O)NC(C2CC(NC(=O)C(C3CCOCC3)C)C2)C)cnc1C C(=O)(C(C)(C)C(C)(C)O)NC(CNC(C1N(CCC)CCC1)=O)C1CC1 Cn1ccc2cccc(C(N3CCCC3CC(=O)N=c3cc(Cl)[nH][nH]3)=O)c12 C1(NC(Cc2cc(OC)c(O)cc2)=O)CCCC12CN(C(=O)Cc1cc[nH]n1)C2 Cn1c(C(=O)NCC23CC2CN(C(c2csc(-c4ncc[nH]4)n2)=O)C3)cnc1O C(=O)(CC1COc2ccccc21)NC(CC1CCN(C(C=CC)=O)CC1)C c1(C(NOCCOCC)=O)cc(CNC(=O)CC2CSCCO2)nn1C c1(C(N(CCCCCCNC(CC2C(OC)CC2)=O)C)=O)cnc2sccc2c1 C1(C(=O)NCC2N(C(C34CC(F)(C3)C4)=O)CCC2C2CC2)CCn2cnnc2C1 CC1CC(N(C)C(C2CCCN(Cc3cnn(C)c3)C2)=O)CC(C)C1 N1(C(c2c(NC)nsn2)=O)CCC2(CCCC2C(N2CCC(C(=O)OC)C2)=O)C1 c1(NCCOc2cc(C)nn2C)nccc(=NC(CCO)c2cccc(Cl)c2)[nH]1 C1(NC(=O)CN2CC3CC3C2)CN(C(=O)C=C2CCOCC2)CC1C1CC1 C(=O)(CCC(=O)c1ccc[nH]1)N1C(CNc2ccc(C(C)(C)C)cn2)CC1 C(=O)(CC1=CCCCC1)N1CCC(O)(CCNC(C2(C)CC=CC2)=O)C1 c1(C(=O)NC2(CC)CN(C(=O)C(CC3CC3)OC)C2)cc2cccnn2c1 C(C(F)C(=O)N1CC(C(=O)NCC2(OCC)CC(C(F)(F)F)C2)C1)N(CC)CC C(=O)(C(C)CC(F)F)NCC1CCC(NC(c2n(C(C)C)ncc2Cl)=O)C1 n1(CC(=O)NCC(CO)NC(C2(F)CCS(=O)(=O)C2)=O)ncn2nccc2c1=O Cc1cc(C(=O)NCC2CCCCN2C(C2CCC(C)C(C)C2)=O)ncc1N C1(CN(C(=O)C=CC2CCC2)C)CCCC1NC(C1(CCNC(N)=O)CCC1)=O n1(CC(=O)NCC2CC2C(=O)NCC(CO)C2CCC2)cc(Cl)cn1 N1(CC(=O)NC2CC(F)CN(C(=O)CC3CCCC3)C2)CCCCCCC1=O.CC c1(C(=O)NCC=CCNC(CCN(CCC(C)(C)C)C)=O)c[nH]ccc1=N N#CCCCCC(=O)N1CCC(CNC(C2CCC3CC3C2)=O)CC1 Cc1ccc(C(=O)NCC2CCCC2NC(c2c(Cl)n[nH]c2C)=O)c(N)c1 C1(OC)CC2CC1CN(C(C1(F)CCN(C(c3c[nH]c(=N)o3)=O)CC1)=O)C2 c1(C(=O)NC2C(F)CCN(C(C3C(C)CC3)=O)C2)cc(=O)c2ccccc2n1C CC1CN(C(c2cc(CNC(=O)CC=C(Cl)Cl)[nH]n2)=O)C1(C)C C1(NC(c2ncc(NC)nc2)=O)CC2CC(NC(c3cc(F)c[nH]3)=O)CC12 C1(CNC(=O)C(F)C(F)(F)F)CC2(CO1)CN(C(c1ccn3nnnc3c1)=O)C2 c1(NC(=O)NC(c2ccncc2Cl)C)ccc(N2CCNC2=O)cc1 c1(C(N2CCCC(N(C(c3cnc(NC(C)=O)o3)=O)C)C2)=O)ccc(N)cc1O c1(OC)ccc(C2(C(=O)NC3CC3CNC(=O)CC3CCSCC3)CC2)cn1 c1(-c2nc(-c3cc4cc(C)ncc4cc3)nn2C)cc2c(cc1F)NC(=O)CC2 C(=O)(CCCC(F)(F)CO)NCC1N(C(c2c(OC)ccc(OC)c2)=O)CC=C1 C1(c2c(OC)ccc(F)c2)CN(N2CCC3(CCNC(=O)N3)C2)CCO1 c1(C(=O)NC(C)CN(C)C(C23CSCC2C3)=O)cnc(C(F)F)nc1 c12ccc3c(c1)CN(C3)Cc1cccnc1-2.c1(OC)ccc(Cl)c(C(=O)N(C)C)c1 Cc1ncc(C(=O)N(C)CC2CCCN2C(=O)C(C)c2ccon2)cc1N c1(OC)cc(Br)c(Cl)cc1C(N1CCN(C(C#N)C(C)(F)F)CC1)=O c1(COC)cc(C(=O)NCC2OCCC2C(=O)NC2CCOC2C)n[nH]1 N#Cc1ccc(C(N2CCC(=CC(=O)N(CCCO)C3CC3)CC2)=O)c(Br)c1 C1(N(C(C=C2CCC(C)C2)=O)C)CCC(NC(C2CC(C)(C)CO2)=O)CC1 C1(C(N(C2CCN(C(=O)CCc3c(C)noc3C)C2)CC)=O)CCCS(=O)(=O)N1 Cc1cc(C(=O)NCCCN(C(=O)C=Cc2cncc(O)c2)C)nc(C)n1 C(=O)(C(C)(C)CCC(=O)OC)N1CCC(C2(NC(C(CC)OC)=O)CC2)C1 C1(C(=O)NC2C(NC(c3cc(SC)nn3C)=O)CCC2)CCn2cncc2C1 CC(C)(C#Cc1cn(CC2CC3CCC2C3)nn1)NC(=O)CC1COCCOC1 c1(C(N(CCNC(C2C(OC)C2)=O)CC2CC2)=O)ccc([N+](=O)[O-])c(NC)n1 CCC(O)C(C)C(=O)N(C(C)CN(C)C(C1(C(=O)OC)CC2(CCC2)C1)=O)C CC(C(=O)NCC1CC(O)CN1C(=O)Cc1cnc[nH]1)C(C)(C)c1ccccc1 N1(C(Cc2c(C)nccc2)=O)CCC2(NC(c3cnn(C)n3)=O)CCCCCC12 CC(C)C(C)C(=O)N1CCC1C(C)(C)NC(=O)CC1(N(C)C)CC1 c1(C(=O)NCCC23CCC2CN(C(C2CS(=O)(=O)C2)=O)C3)cc2ccccc2s1 N1(N(C(C)=O)C2CC2)CCC(C)C(C)C1.c1(N)ccc(NC(=O)CCF)cn1 C12(C(=O)NCC3CCC(NC(C(C)=CCO)=O)C3)OC3C4C5CC(C6C5C3C16)C24 c1(CCC(=O)NC2CC2CNC(C2(Cl)CC2)=O)ccc(Cl)s1 C(CC(C(=O)NCCn1ccnn1)NC(=O)CC(CC)N(C)C)=CC N1(C(C2OCCN(CC)C2)=O)CC2OCCN(C(c3cn(C)ccc3=O)=O)C2C1 C(=O)(C(CC=C)CC(C)C)NC1CCN(C(c2ccc(C#C)cn2)=O)C1 N1(C(C=Cc2ccc(C)s2)=O)CCCC(NC(=O)C(C)N2CCCC2)C1C CC(C)(C)CCCCC(=O)NCC1CC(NC(C2CCOCC2(C)C)=O)C1 O=C(CC1=CCC(NCc2csc3cc(Cl)ccc23)CC1)NC(=O)C(F)(F)F c1(C(=O)NCC2(C)N=C(C)SC2)cnc(Cl)c(C)c1 Cc1cc(S(N)(=O)=O)cc(C(=O)NCC=CCNC(=O)Cc2csc(=N)[nH]2)c1C N1(C(COc2cc(C)on2)=O)CC(C)(C)OCC1CNC(=O)C(O)CCN(C)C N1(C(c2nn(C)c(Cl)c2)=O)CC(NC(C2CCCCC2C(N)=O)=O)CC12CCC2 c1(C(=O)NC(C(C2CC2)OC)C)cncc(C)c1.C1(NC(=O)C2CC2)(CO)CCCC1 c1(OC)ccc(C(=O)N(C)CC2CC(F)CN2C(C2CC(F)CN2C)=O)nn1 N1(C(C(CCC)O)=O)CCN(C(=O)CCc2ccc(O)nn2)C(CCC)C1 NC1CC2CC2C(CNCC(N2CCc3ccccc32)c2ccc(Cl)cc2)C1O c1(OC)ccc(Br)c(CNCC2COCCOC2)c1F c1(C(C(=O)OCC)N(C)Cc2ccc(OC)c(Cl)c2)cccc(Br)c1C N1(C(CCCCC=C)=O)CCC(NC(c2ccnn2CC#N)=O)C(F)(F)CC1 CC(C)S(=O)(=O)C(C)C(=O)NCCN(C(c1cc2cccnc2s1)=O)C1CC1 N1(C(c2cccc(C(F)F)n2)=O)CC(NC(C2(O)COC2)=O)CC12CCCOC2 c1(NC(=O)C(Cl)(Cl)Cl)ccc(NC(C2CC(CC3CC3)C2)=O)cn1 C(=O)(C1=COCCC1)NC(C)CC(=O)N(C1CCNC1=O)C C(=O)(C1=CCC2CCC1N2C(C1CCC(C2CC2)C1)=O)N1CC(C(C)C)OCC1 c1(C(=O)NCC2CCN(C(C3C(C#C)C3)=O)C2(C)C)c(C)nn2cc(C)cnc12 S(=O)(=O)(c1cnc(NCCC2CCCC2)c(Cl)c1)NCCS(C)=O N1(C(C(C=CC)O)=O)CC2CC(C1)C(CO)C2NC(c1cc(C)c(N)cc1Cl)=O N1(C(c2c(C)ccc(Br)c2)=O)CC2CCN(C(c3ccnc(C(F)F)c3)=O)C2C1 N1(C(C(C(CC)C)C)=O)Cc2nccn2CC(NC(C2CC23CC3)=O)C1 N1(C(C2=CCCC2C)=O)CCN(C(c2ccc(C(N)=O)cn2)=O)C2COCC12 c1(CCC(=O)NC2(CF)CCN(C(CC3CC(=C)C3)=O)C2)ccc(Cl)c(Cl)c1 C1(CC)CCN(C(=O)Cc2cccnc2F)C1C(=O)NCC(F)(F)C(N)=O N1(CCOCC=C)CCC2(CN(C(c3sccc3OC)=O)CC(C)O2)C1 C1(C(=O)NC2CC(CCC(=O)NC(CC)C(=O)OC)C2)CCC(O)CN1C c1(CC)nocc1C(N1CCOCC1)C(=O)NC(C)(C)CC c1(C(=O)NC(C2(c3cccnc3)CC2)=O)cccnc1N1CCC(N(C)CC)C1 C(=O)(C(CNC(=O)CSC(C)(C)C)C(C)(C)C)N1C(C=C)CC1 C(c1ccc2c(c1)CCO2)=CC(N1CCN(C(C2C(C)CC2)=O)C(C2CC2)C1)=O [N-]=[N+]=NCCCCCCC(=O)NC(CNC(C1CCOC2(CCC2)C1)=O)C1CC1 Cc1cccc(NC(C2CCN(C(=O)CC(c3cccc(F)c3)O)C2)=O)c1 N1(C(c2ccc(CC)o2)=O)CCC2(CC1)CC2CNC(C1(CC(C)C)COC1)=O N1(C(C=Cc2cccc(OC)c2)=O)CCN(C(=O)CCNC(C)=O)CC1C#N C(c1cccc(CO)c1)=CC(N1CCCC(N(C(=O)Cc2cncs2)CCO)C1)=O N1(C(=O)Cc2ccc(Cl)c(Cl)c2)CC(C2CN(C(C3CCC(F)C3)=O)C2)C1 N1(C(C2(CC)CC2)=O)CC(F)(CNC(c2ccc(-c3csc(C)n3)s2)=O)C1 C1(NC(c2cnsn2)=O)CC(O)CN(C(c2cn[nH]c2)=O)C1 C1(NC(C2C(C)CC2)=O)CCC(NC(c2cnc(Cc3ccccc3)s2)=O)CC1 C1(COC)(NC(c2cncc(Br)c2)=O)CCN(C(C2CC2C#N)=O)C1 C#Cc1ccc(OC)c(C(=O)NCC2CCN2C(c2cnc(COC)o2)=O)c1 C1(C(=O)NC(CC#C)C(=O)OC)CCN(C(=O)CCc2ccccn2)C1(C)C C1(NC(C2N(C(C)=O)CCOC2)=O)CN(C(=O)CC2CC(C)(C)C2)C(C)(C)C1 C(C)(CC(=O)NC1CC(NC(=O)Cc2cn[nH]c2)C1)OC C1(C(N(C)C)=O)CCCCN1Cc1ccc(=N)[nH]c1 N1(Cc2n(C)ccc2)CC2C(C1)N2C(=O)CNC(c1ccc(F)cc1)=O C=CC(C)(C)C(=O)N1C(C(=O)NCC2CCC(F)C2)CC2CC12 c1(C(N(CC(C)NC(C2N(CC)CCC2)=O)C)=O)ccc(O)c(C(C)(C)C)c1 C1(CC(=O)N(CC(C)N(C(=O)C(O)CC2CCCC2)C)C)CCC(C)(C)O1 c1(C(=O)NCC2(O)CN(C(c3cc(OCC)ncc3)=O)C2)ncc2ccccn12 S(=O)(=O)(c1ncccc1Br)C(=O)NC1(C)CCCC(F)(F)C1 Cn1nc(C(=O)NC2(CCO)CN(C(=O)Cn3cnc(C(F)(F)F)n3)C2)cc1O N1(C(Cc2cc(C)no2)=O)CC2CCN(C(=O)CCc3cccnc3)CC12 C1(CC(=O)N(CC=C)CCNC(=O)CCSC(F)(F)F)(C(=O)OC)CCCC1 Cc1cc(Cl)ccc1CC(N1CCCC(O)(CCNC(=O)C(C)CN(C)C)C1)=O C1(C(N2CCC(C)(C(=O)OC)C2)=O)CNC(=O)CN1C(C1CCC1C)=O C1(NC(c2cc(Cl)ccc2O)=O)CC2(CCCCN2C(c2ccccc2)=O)C1 CC1CN(C(=O)OC(C)(C)C)CC1N(C1(c2cccs2)CC1C)C(C1CCC1)=O CCCCC(O)C(=O)NC1(C(N2CC(C)(N(C)C)C2)=O)CCC1 C(=O)(C1=CCCC(C)(C)C1)NC(C1CCCCC1)CNC(c1c(C)nc(C)o1)=O c1(CC)nc(O)sc1S(=O)(=O)N(C)Cc1ccc(C)cc1Cl S(=O)(=O)(c1ccccc1Cl)NCC(N1C(CNC(C(C=CCCC)O)=O)CC1)=O c1(C(=O)NC(CCN(C(C(CC)CC)=O)C)C(C)(C)C)c[nH]c2cnccc12 c1(C(N2CC(CN(C(c3cc(C)ncn3)=O)C)OCC2)=O)cc(O)nc(O)c1 C1(NC(CSc2n[nH]c(=N)s2)=O)CC12CCC(NC(c1ccc(Cl)o1)=O)CC2 CC(O)(CC(F)(F)F)C(=O)N1CC(CNC(=O)CN2CCN(C(N)=O)CC2)C1 c1(C(C)C)cncc(C(=O)NCC(CO)NC(=O)CNC=O)c1 C1(NC(C=C(CC)CC)=O)CC2CCC(C1)N2C(C1CC2OC1C1CC21)=O CC1(C)CCN(c2nnc(-c3ccccc3N3CCCCC3)n2CC2CC2)CC1 O=C(CNC(N1CCN(c2ccc(F)cc2)CC1)=O)NNc1ccccn1 CC12CC(CC(=O)NCC3(NC(c4c(Br)ccn4C)=O)CC3)(CO1)C2 N1(C(C(=O)NC2(c3nc[nH]n3)CCCC2)C2CC2(Br)Br)CC2CC2(CO)C1 C12(C(=O)NCCCN(C(c3cc(C(F)F)no3)=O)CC)CC3CC1C2C3O N1(C(C(C)n2cnnn2)=O)CCC(NC(c2cccc(C(F)F)n2)=O)CC(O)C1 c1(CSC)cc(C(=O)NCCCNC(=O)C(C)N(C)C(C)=O)c(C)o1 Cn1ccnc1C(C(=O)NC(C)(C)C)N(C)C.C1(C)(C)CNC(=O)C2(CC2)C(=O)N1 Cc1cc(C(N2CCCC(CN(C(=O)CC3(C)OCCO3)C)C2)=O)cc(Cl)c1 C1(N(C)C)CCCC(N=c2[nH]c(N3CC4(CCCN4C)C3)nc3ccsc23)C1 N1(C(CCOCCC)=O)CCN(C(c2cc(C3CC3)nn2C)=O)C(C)C1C CC(C)CC(C(=O)NC1C2CCC1N(C(C1CCS(=O)(=O)CC1)=O)C2)NC(N)=O N1(C(c2cccc(OCCC)c2)=O)CCC(C)C(NC(=O)C(F)=C2CCC2)C1 C12CCC(CC1)C(=O)N2.N1C(=NCC2CC2)NC2CCCC2C1.CCOC c1(C(=O)OCc2c(OC)c(F)ccc2)cc(S(=O)(=O)Cc2cccnc2)ccc1F CC(C)C(C(=O)OC(C)(C)C)C(=O)NCCC(O)CNC(=O)Cc1nnc(O)s1 Cc1cc(Cl)cc(C)c1C(=O)NCC12CCC1CCN2C(c1nc(=O)n(C)[nH]1)=O CC1OCCC1CC(=O)NC(C)(C)C(=O)NCCN1CCC1 c1(N(CCC)C)nc2cc[nH]c2c(=NCC2CCc3cc(F)ccc3O2)[nH]1 C1(C(=O)NCCCC2N(C)CCC2)CCCN1NC(=O)CCC1CC1 C1(C(=O)Nc2ccc(C(N)=O)cc2)CN(C(c2cc(O)ncn2)=O)CCC1O C1(C(=O)Nc2ncccc2I)CN(C(c2cc(Br)ccn2)=O)CCC1O CCCC(C(=O)NC1CC(NC(=O)COc2cccc(OC)c2)C1)N(C)C N1(C(C2N(CC)CCC2)=O)CC2CC1C2CNC(=O)CCc1cc(Cl)no1 N1(C(c2cnc(CC)nc2)=O)CCC(C(=O)NCCC2CCN(C)C2=O)C1(C)C c1(C(=O)NC(CN(C(=O)Cc2cccs2)CC)C)cn(C(F)(F)CO)nn1 CC(C)CC(CNC(C1(C(F)(F)F)CCCCC1)=O)NC(C1(C)COC1)=O c1(C(N2CCCCC(N(C)C(c3cccc(Cl)c3)=O)C2)=O)ccccc1S(C)=O c1(C(=O)Nc2cnc(C(F)(F)F)cn2)c(F)cc(Cl)cc1Br.C1(C=O)CC1 c1(CCCC(=O)NCCOCCCNC(C2C(C(N)=O)CC2)=O)ccccc1Cl c1(COC)nc(NCCCC(F)F)cc(N2CCCC(CCCO)C2)n1 c1(Cc2cn(CC3CC(CNC(C4CCC(=O)N4)=O)C3)nn2)cccc(Cl)c1 O=C1Cc2cc(C(N3CC4CCN(C(=O)C5=COCCC5)CC4C3)=O)ccc2N1 C1(C(C)NC(C2(F)CC2)=O)CCN(C(=O)CCC2CCCC(O)C2)CC1 C1(NC(=O)C2=COCC2)C2CC(O)C1N(C(c1cncc3ccsc13)=O)C2 c1(OCCC(N2CCN(C(c3ccncn3)=O)C(CO)C2)=O)ccc(F)c(Cl)c1 c1(C(C)(F)F)n[nH]cc1C(=O)NC1(C)CC(NC(C2CN(CC(F)(F)F)C2)=O)C1 C1(OC)(OC)CCSCC1NC(=O)NCc1cnc2sccn12 C1(C(N2CC(N(C(c3n(CCOC)ncc3)=O)C)C2)=O)C2CC3C(C2)C13 N1(C(CCN(C(=O)C(C2CCOC2)OC)CC)=O)C(C)CCCC1C Cc1ccc(C(N)=O)cc1C(=O)NC1(C2CN(C(=O)CCC(F)F)C2)CC1 N1(C(C(F)=C(C)C)=O)CC2CC1CCN2C(=O)CCc1ccncc1Br C(=O)(C(C)(C)CC#N)NCC(CNC(c1cccc(CCC)c1)=O)F C1(C(=O)NC2CC=C(C)CC2)C2CCC(C2)C1C N1(C(c2ccc(N)cn2)=O)CCC(NC(=O)C=Cc2ccncn2)C(F)(F)CC1 C(=O)(C1CCCn2ccnc21)NC1CN(C(C(C)OC(C)=O)=O)CC(F)(F)C1 N1(C(C=CC=CCC)=O)CC(NC(C2(CF)CC2(F)F)=O)C(C)C1 CC1CCN(C(=O)C(c2ccc(F)cc2)(C)C)CC1NC(C1(CO)CCCO1)=O C1(C(N(CC(=O)N(C)C)CC)=O)CN(C(=O)C(C)OC(C)=O)CCC1(C)C c1(-c2nc(C(CC)C)nn2C(C2(C)CC2)C)ccc(F)c2occc12 C1(C(=O)NCC2(C)COCCN(C(CCS(C)=O)=O)C2)CS(=O)(=O)CC12CCC2 n1(CC)nc(C)c(CC(=O)N(C2CCS(=N)(=O)C2)Cc2ccccc2Cl)c1C C1CCC(C)C1.C1(C(=O)OC)CC(C(C)C)C1.C1C(=O)N1CCOC C(CC(C)C)(C(=O)NC(C)Cc1cc(C)[nH]n1)NC(c1cc(CC)sn1)=O Cc1cccc2c1OCCC2NC(N1CC(c2ccoc2)CC1C)=O c1(OCc2nnc(N(CC#C)CC=C)n2CC2CCOC2)ccc(C)cc1C C1(CNC(COCCOC)=O)CCCC2CN(C(=O)C(C(C)C)N(C)C)CC12 c1(C(=O)NC2C3CN(C(C(CC)(F)F)=O)CC32)cc2c(s1)CCSC2 CC(Cc1ccc(Cl)cc1)CC(=O)OCCSCC1(O)CC1 N1(C(C=CC(C)=O)=O)C2CCC1CC(CNC(C1CC(C(C)(C)C)=NO1)=O)C2 c1(C(=O)NC(c2cn(-c3ccc(Cl)cc3F)nn2)C)cnn2cccnc12 c1(CC)nc(C)[nH]c1C(N1CCC(CNC(C2OCCOC2C)=O)C1)=O C1(NC(c2cc(O)cs2)=O)CC2CC(NC(C3C4COCC34)=O)C1C2 Cc1cnc2cccc(C(=O)NCCC3CCCN3C(c3nc(=O)n(C)[nH]3)=O)n12 C(=O)(CCCCCN=[N+]=[N-])N1CC(C(=O)NCc2nc(CC)[nH]n2)(C(C)C)C1 C(N=c1[nH]c(N(C)Cc2ccnn2C)nc2c1CCCC2)c1cc(OC)nn1C c1(OC)ccc(C(N2CCOCC2CNC(=O)C(C)CSC(F)(F)F)=O)c(O)c1 c1(CC)cc(C(=O)NCCC2CCCN(C(=O)C(F)CC3CCCC3)C2)ncn1 N1(C(c2cc(C)sc2)=O)CCC(F)(C(=O)N(C2CC(C)CC(C)C2)C)CC1 CC1=NOC(C)(C(=O)NC2CCN(C(C3CCCCN3S(C)(=O)=O)=O)CC2)C1 C(=O)(CC(C(C)(C)C)NC(c1csnc1C)=O)NC1CN(CC)CC1C c1(CNc2cn(C)c(C(=O)Nc3cnn(C4CC4)c3)n2)ccc(Br)c(O)c1 N1(C(CC2(C(=C)F)CCC2)=O)CC(CNC(c2ccnn2CCC)=O)C2(CC2)C1 C1(C(N2CCCC(NC(C(C(C)C)=O)=O)C2)=O)CCC(O)CN1C C1(CNC(C=CS(C)=O)=O)CCCCN(C(c2cc(-c3ccco3)on2)=O)CC1 N1(C(Cc2nc(C)sc2)=O)CCN(C(=O)C=CC2CCC2)CC(C)(C)C1 c1(C(N2C(C3CCN(C(C(C)C)=O)C3)CCCC2)=O)ccc2oc(=O)oc2c1 C=C(C)C(C)(O)C(=O)NC1CCN(C(=O)COc2ccc(Br)c(C)c2)CC1 c1(C(N2CCC(O)(CN(C(c3c(C)nns3)=O)C)C2)=O)cccc2c1OCC2C CC(C)C(C(=O)N(C)CCNC(c1cn(C)[nH]c1=N)=O)NS(=O)(=O)C1CC1 c1(NC(c2scc(CNC(COC(CC)(C)C)=O)c2)=O)cc(C)cc(C)c1 C1(NC(CCSC)=O)(CNC(=O)C(c2ccc(C)o2)C)CC2CCC1CC2 C(=O)(CCC(C)O)NCCC1N(C(CC2ON=C(C)C2)=O)CCC1 c1(OC)cc(NC(c2cc(Cl)cc(Br)c2)=O)c(-c2cc(O)ccc2F)cn1 C=CCC(CNC(c1cnn(C2CC2)c1)=O)C(=O)N1CCOC(C)C1CO c1(C(=O)NC(COC)CNC(C2CCCOC2C)=O)ccc2nnc(C)n2c1 C1(C(=O)NCC(C(=O)OCC)C)(CF)CCN(C(=O)CC2CCSC2)C1 C(C)(CNC(=O)CC1CCC(C)(C)CC1)(CC(C)C)NC(COCCOC)=O c1(C(N2CCC(NC(C(CC#C)C3CC3)=O)C2C)=O)cc(F)ccc1C#C c1(OC)ccc(C(N2CC3C(C(=O)N=c4[nH]nc(Cl)cc4C)C3C2)=O)cc1[N+](=O)[O-] C(C)(N=c1cc(C)nc(N2CCn3nc(C)nc3C2)[nH]1)c1ccc(OC)cn1 N1(C(C=C(C)Cl)=O)CC2CC3CC2C1C3NC(c1n[nH]c(C)c1C)=O c1(OC)ccc(Br)c(NC(C2CC2C(=O)N(C)CCc2ccccc2)=O)n1 N1(C(CCN(C)CC)=O)CCCC(NC(=O)CCc2cccc(F)c2F)C(F)C1 C(=O)(CC(O)CCSC)N1C(C(C)NC(CNC(CC)=O)=O)CCCC1 C1(NC(C=C(C)C)=O)CC2CCC1N2C(C1CC1[N+](=O)[O-])=O C1(CCNC(C2(CCCC)CC2)=O)CCN(C(=O)CCCc2cccs2)C1 Cc1ccc(C)c(C(N2CCC(NC(C3CC4(C3)CC4F)=O)C23CC3)=O)n1 c1(C(=O)OCC(CC)OC)ccc(C=CC(=O)O)c([N+](=O)[O-])c1 N1(C(C2C(c3ccc(C#N)cc3)C2)=O)CC2CCC(C1)C2NC(C1CC1F)=O Cc1nc2cncc(C(=O)Nc3c(O)cc(C(=O)O)cc3C#N)c2[nH]1 CC(C(=O)NCCc1cc[nH]n1)NC(=O)C=CC1CCC1 CC1=C(C(=O)NC(C2CCCN2C(=O)CN2CCCS2(=O)=O)C)SCCO1 C1(NC(CN(C)C(c2ccsc2)=O)=O)CCC(NC(=O)CCCc2cncs2)CC1 C(=O)(C(CNC(C1COCC(C)O1)=O)C(C)C)NC(CCOC)C Cc1cnncc1C(=O)NC1CCN(C(=O)C(C(C)C)n2cncn2)C1C1CC1 N1(C(CCC(=C)Cl)=O)CCC(C2CCN(C(=O)CCCc3n[nH]c(=N)s3)C2)C1 C(=O)(CC(C)CCC)NC1(CC=C)CCN(C(c2cc(C)ncc2C)=O)C1 c1(C(N(CCCOCCNC(=O)C(O)C2CCC2)C)=O)nn2cccnc2c1Cl C1(C(=O)NCCC(C)NC(C2(C(=O)N(C)C)CC2)=O)CCCOC1C C1(NCCCC)CCC(N=c2[nH]c(=NC)[nH]c(=NC(C)C)[nH]2)C1 c1(OC)ccc(CNC(=O)NCC2CC(N)C2)c(OC)n1 C1(C)(CNC(C2C(C(C)C)CCO2)=O)CCN(C(=O)CC2CCC3CC23)C1 S(=O)(=O)(c1ccc(F)cc1)NC1CC2(CC(NC(=O)CCCn3cccc3)C2)C1 c1(C(=O)NC2CC(c3noc(-c4cccs4)n3)C2)ccccc1F C(C)(CC(C)NC(C1(COC)CCC1)=O)NC(C=CC=CCC)=O CCCCCCC(C)C(=O)NCC1CCOC1C(=O)NCCn1cnnc1CC C(CO)(CCCCNC(C1(c2ccc(F)c(Cl)c2)CC1)=O)NC(C1C(CC)C1)=O C(C(CO)C(F)(F)F)NC1c2conc21.c1(C(C)(C)C)nnnn1CCCF c1(CC)nn(C)c(CC)c1C(N1CC=C(CNC(=O)Cc2ccno2)CC1)=O c1(C(C(=O)N(C2CC(O)C2)C)NC(CCOCC#C)=O)ccccc1 C1(C(N2CCC(NCc3ccccc3)CC2)=O)CCCN(c2ncccn2)C1 N1(C(C2C(CC)CCC2)=O)CCC(=CCNC(=O)CC2CC(=O)NC2=O)CC1 C1(F)(CNC(C(CC)=CC)=O)CCCN(C(c2ccc(OCC(N)=O)cc2)=O)C1 C(=O)(C1CCCn2cnnc21)N(CC(C)CNC(c1c(F)cnn1C(C)C)=O)C C1(C(N(CC(COC)O)C)=O)CC2(CCN1C(C1COCOC1)=O)CC2 c1(C(N2CC3C(CNC(=O)C=Cc4cnc[nH]4)(C3)C2)=O)cc(Cl)nc2n[nH]cc12 C1(C(=O)NC(C)C(=O)N(C)C)CCCCCC1NC(c1cccs1)=O c1(C(N2CC(OC)(CNC(c3csc(C)n3)=O)C2)=O)cnc(P(C)(C)=O)cn1 C1(CNC(C(c2cscn2)N(C)C)=O)CCCC(NC(=O)C=Cc2ncc[nH]2)C1 C(c1cncc(O)c1)=CC(=O)N(C)CC1(NC(=O)C=Cc2cocn2)CC1 C1(CC(=O)NC)CN(C(C2CCCN2C=O)=O)CCN1C(c1cc(C#N)c[nH]1)=O N1(C(=O)Cc2cc[nH]n2)CC2CCC1C1CN(c3nccn4nnnc34)CC21 c1(C(C)C)ccc(C(=O)NC2CCCN(C(c3ccccc3F)C)C2)cc1Cl c1(C(=O)NC(C(=O)N(CCCC(C)O)C)COC(C)C)ccc2n[nH]cc2c1 C1(C(=O)NCC2CC(CNC(=O)CC=C(Cl)Cl)C2)CC2(COCCO2)C1 C(=O)(CCC(F)(F)F)NCC1CCC(NC(c2[nH]cc(CC(C)C)c2)=O)CC1 C1(C(=O)NC(C)CCc2cn[nH]c2)C(C2CC2)CCN1C(=O)CC(C)(C)C#N C(CNC(C1(C)CC(F)(F)C1)=O)(C(C)(C)C)NC(Cn1ccc(C(=O)OC)n1)=O c1(C(=O)NCCC2CCCN(C(c3n[nH]cc3Br)=O)C2)cc2n(c1)CCC2 C1(OCC)CC2CN(C(=O)C(COC)NC(c3c[nH]nc3CC)=O)CC12 C12(C(=O)NCC(C)O)COC(C1)C(NC(C1CCC(C)(C)CC1)=O)C2 n1(CC(=O)N(C)CC2CN(C(C3CCCC3O)=O)C2)ccc2ccc(F)cc12 C1(C(=O)NCCN(C(c2ccc(C(C)C)o2)=O)C2CC2)Cc2c(F)cccc2O1 N1(C(C(C)NC(=O)CC(C)C2CC2)=O)CCN2CCCCC2C1 C1(C2CCCN(C(=O)C(CCc3ccccc3)CC(C)C)C2)(C(=O)OCC)CC1 C(C(C)(CC)NC(=O)CC1CC=CCC1)NC(CNC(=O)OC)=O Cc1[nH][nH]c2ncnc(=NCC3CC(NC(c4cc(Cl)sc4Cl)=O)C3)c1-2 C1(SC)(CN(CC(C)(C)OC)C(=O)OCCCC(C)C)CC2CCCC12 N(C(=NCC1CCCC(C(N)=O)C1)NCc1ccccn1)C(CC)CC c1(SC(C(N2CC(C)(NC(Cc3c(C)n[nH]c3C)=O)C2)=O)C)ccc(F)c(F)c1 C1(O)(C(C)NC(CCOC(C)=O)=O)CCN(C(=O)Cc2ccccc2CO)CC1 C(C)(c1ccccc1Cl)=CC(=O)NC1CC(NC(c2[nH]cc(C(C)=O)c2)=O)C1 Cc1cccc(C2CC(NC(C3CC3c3ccccc3C(F)(F)F)=O)C2)c1 Cc1cccc(CNC(=O)CC2CCCN(C(C34CCC(CC3)CO4)=O)C2)c1F C#CC1CN(C(c2coc(CC)n2)=O)CCN1C(c1cc(C)c(F)cc1N)=O CCCC(CCCNC(C1CC(NC(c2ccn(C)c2)=O)C1)=O)NC(=O)CSC Cc1c(C(=O)Nc2cc(F)c(N)cc2Cl)oc2c(Cl)cccc12 C12(C(=O)NC(C3CN(C(c4n(CC)ncc4)=O)C3)=O)CCC(COC)(CO1)C2 C1(C(N(CCC(=O)OC)CC)=O)CN(C(c2c(C)csc2C)=O)CCN1C c1(C(=O)NCC2N(C(c3c(COC)cco3)=O)CCC2)ccc(C(F)F)cc1F c1(NC(=O)CC2CN(C(C3CC3(F)F)=O)CCO2)cccc(Cl)c1[N+](=O)[O-] C(=O)(CC(O)C(N)=O)NCc1c(Cn2cc(CCN(C)C)nn2)nco1 c1(OC)ccsc1C(=O)N(CC(C)O)CCNC(C1(C2CCCCO2)CCC1)=O C#CC(CNC(C1CCCCCN1C(c1cc(CC)no1)=O)=O)CC(C)(C)C C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC(CC)CN(C(=O)C(F)OC)CC C1(NC(c2nc(COC)sc2)=O)CC(CNC(=O)CC(C)n2cccn2)C(O)C1 C12(CCN(c3cncc(C(=O)O)n3)CC1)C(=O)N2.c1(CC)cccc(F)c1 CC(C)(F)C(=O)N=c1ccn(CC2CCCO2)[nH]1 c1(CC(=O)N(CC(C)NC(C2CC(N3CC(O)C3)C2)=O)CC)ccc(Cl)cc1 Cc1cc(CN2CCC(O)C(C(=O)NC3CN(C(N)=O)C3)C2)cc(O)c1 N#CCCCCCC(=O)NCC1CC(CNC(c2ccc([N+](=O)[O-])s2)=O)CO1 C1(C(=O)NCc2snc(CC)n2)CCN(C(=O)C(C)SC(C)C)O1 CC1(C)CC(NC(c2cccnc2S)=O)CN(C(c2nocc2Cl)=O)C1 C(C(C(C)C(C)C)NC(c1sc(OC)nc1Cl)=O)NC(c1cnc(OC)s1)=O C(=O)(C1=CC2CCC(C1)C2)NCC(CC(C)C)C(=O)NCCC(=O)NC(C)C S(=O)(=O)(CCC(=O)NCCC(C)N(C)C(C1CCOC(C)(C)C1)=O)NC C1(NC(c2cccc(-n3ccnc3)c2)=O)C2CC(O)C1N(C(=O)C1=NOCC1)C2 c1(C(=O)OCC)cc(Br)c(S(=O)(=O)NC(CN)C(=O)OC)cc1C Cc1cc(CNC(=O)CCC2(NC(C34CCC3C4)=O)CCCC2)cc(C)n1 C1(NC(CCN(C(CC)CC)C)=O)(CO)CCCN(C(=O)Cc2cnc[nH]2)C1 N1(C(C(C)(C)C(F)F)=O)CC2CCCC(C1)N2C(=O)CSCc1ccc(Cl)cc1 c1(C(N(CCN(C(c2n[nH]c3c2COC3)=O)CC)CC)=O)ccc(S(C)(=O)=O)s1 Cc1cnc(C(=O)NC(CN(C(=O)C2=CCSC2)C)Cc2ccccc2)cc1Cl C1(C(C)C)CN(C(C2CC3(CCC3O)C2)=O)CCN1C(c1ccc(Cl)cc1Cl)=O CC(C)CC(O)C(=O)N1CC(F)(C(=O)Nc2ccc(O)cn2)C1 c1(C(=O)NC2C(C)CN(C(=O)CSCCC(F)(F)F)C2)cc(F)c(O)c(F)c1 c1(C(N2CCC3(C(C(=O)Nc4cc(C)cc(Br)c4)C3)C2)=O)cnc2ccccn12 CC(C)(C(=O)N1CCOC2(C1)CN(C(=O)C(F)C1CC1)C2)C1=CCSCC1 C1(C)(CNC(C2(N(C)C)CCCSC2)=O)CN(C(c2cnn(C)n2)=O)CCO1 N1(C(c2cnc(C(C)C)[nH]2)=O)CC(CNC(c2cc[nH]c2C(C)C)=O)CC1C C#CCC(C)C(=O)NC1(c2ccccc2)CC(NC(=O)C(C)C=C=C)C1 N1(C(CCc2n(C)ncc2)=O)CCC2C(CCCN2C(C2CCCC2O)=O)C1 Cc1cnc(CC(=O)N(CC(C)C)Cc2nncn2C)[nH]1 c1(C(=O)NC(c2nccs2)CC)n[nH]cc1CNC(=O)C(c1ccn(C)n1)C Cc1nc(S(C)(=O)=O)sc1C(N1CC(CO)C2(C1)CN(C(C1(C)CC1)=O)C2)=O N1(C(C(C)N(CC)CC)=O)CCOCC(C(=O)NC2(CF)CCCC2)C1 C(=O)(C#CC(C)(C)CNC(=O)C(c1ccnn1C)O)NCCCCOC C1(C(N(CC(O)CN(C)C(C2CC(=O)OC2(C)C)=O)C)=O)C2CCC1(C)C2(C)C CC1(C)OCCOC1CC(=O)NC1CCCOC1 c1(CNC(=O)NC(C(CC)C)C)c(C)nsc1C c1(C(=O)NC2CC(C)(NC(=O)CCc3ncc[nH]3)C2)ccc2c(c1)COB2O c1(NC2(c3n(C(CC)(C)C)nnn3)CCSC(C)C2)cnc2n1CCCC2 N1(C(C(=O)Nc2cc(C)c(N3CCNC3=O)cc2)=O)CC(C2CCC2)C1C(=O)OC Cc1[nH]nc2c1CC(C(N1CCC(NC(=O)C=CC(=O)OC(C)(C)C)C1)=O)CC2 N1(C(C2(SC)CC2)=O)CC(C)C(NC(=O)COCc2cccnc2)C(C)C1 CC(C)S(=O)(=O)C(C)C(=O)N1CCC(C)(C)C(NC(=O)Cc2csnn2)C1 n1(CC)cc(CC(N2CCCC2CC(=O)NCC(C2CCCC2)C)=O)nn1 N1(C(C(C)=CC)=O)CCOCC1C(C)NC(c1csc(COCCOC)n1)=O Nc1nn2ccccc2c1C(N1CC2C(NC(C3CCCCC3)=O)C2C1)=O C1(C(=O)NCC2(CC)CN(C(C3(COCC)CC3)=O)C2)C=CC=CC=C1 C1(C(=O)NCC(C(C)(C)C)NC(c2cccnc2O)=O)CN2CCN1CC2 Cc1cc(C(=O)O)ccc1CN.c1(C)cnc(N2CCCCC2CCO)nc1 c1(C(N2C(C)(CC(=O)NC(c3cn(C)nc3)CO)CC2)=O)ccc(C#N)cc1 C1(NC(c2n[nH]c(C)c2O)=O)CC2CCCC(C1)N2C(=O)CCN1CCCCC1 C(=O)(CC(C(=O)NCC1CN(C(C2CC3CCC2O3)=O)CCO1)NC(C)=O)OC CCC(C)CCCC(=O)NCCCN(C(c1ccc(F)c(Cl)c1N)=O)CC c1(C(=O)OCC)cnc(C(N2CC(NC(c3ncc(OC)cn3)=O)C2)=O)cn1 Cc1ccc(C(N2CCCN(C(=O)Cc3cnc[nH]3)CC2C)=O)c(Cl)c1Cl C1(CNC(c2cc(C)on2)=O)C2CCC(C2)N1C(=O)C#CC(=O)N(C)C Nc1c(F)cc(C(N2CC3CC3(CNC(c3cc(Cl)c[nH]3)=O)C2)=O)c(F)c1F C1(NC(c2scc(C)c2Cl)=O)CC2CC(C1)N(C(c1cc(O)cc(O)c1)=O)C2 C#CCCCCC(=O)NC1(CNC(C2CC(O)(C#C)C2)=O)CCC1 c1(C(C)C(N2CCC(N(CCC(F)(F)F)C(=O)C(C)O)CC2)=O)cc(F)ccc1Br N1(C(C(C)=CC)=O)CC2(CCN(C(C3CC3COC)=O)CC2)C1 c1(C(=O)NCC2CCCN2C(=O)Cn2nnc(=O)[nH]2)cc(F)c(O)c(Cl)c1 C(=O)(C1=CNC2=NCCC2=C1)N1C(CN(C)C(C2CC23CCOC3)=O)CCC1 N1(C(c2cc(C(C)(C)C)sc2)=O)CCCC(NC(=O)Cc2cn[nH]c2)C1 C1(C)(NC(CCc2cc(C)on2)=O)CCN(C(c2csc(C)c2N)=O)C1 C(=O)(C(C)(C)CC(F)(F)F)N1CC(OC)(CNC(=O)C(C)C2CCOC2)C1 c1(CC(N2CCCC(NC(C3C4CCN3CC4)=O)C2)=O)noc2ccc(F)cc12 C1(C)(C(N(C(C)CC(F)(F)F)C)=O)COc2ccccc2O1 c1(OCC)ncc(C(N2CCC(O)C2C(=O)NCC2CCCOCC2)=O)cn1 N(C(=NCCC(C)(C)C1CC1)NC1CC1)C1CCN(S(CCC)(=O)=O)CC1 N1(C(CNS(C)(=O)=O)=O)CC(NC(=O)CC2CCSCC2)CC(O)C1 c1(C2C(C(=O)NC(Cn3cc(C(CC)CC)nn3)C)C2)ccccc1Br C(=O)(C(C)(O)C(C)C)N(C)CC1(NC(CNC(C(CC)CC)=O)=O)CC1 Cc1occc1C(=O)NCC1OCCC1C(=O)NCCc1nc[nH]n1 N1(C(COCc2cc(C)no2)=O)CCC(NC(=O)C(C2(O)CCCC2)C)C1(C)C CC(C)C(C)(C)C(=O)NCCC1(O)CN(C(c2ccc(CS(N)(=O)=O)cc2)=O)C1 c1(C(N2CCC(C3C(C)(C)CN3c3ncc(Cl)cn3)CC2)=O)cc[nH]c(=N)c1N c1(C(=O)NC2CC2C(=O)Nc2cnn(C3CC3)c2)cc(F)c(Br)c(F)c1 CC1c2c(Br)ccc(F)c2CCN1C(C1CCc2cc(N)ccc2O1)=O c1(C(=O)NCC2(NC(c3cc(C(C)=O)sc3)=O)CCC2)c(F)ccc2[nH]ccc12 c1(C(=O)NC23CN(C2)C3)nc(CC)ncc1NC.CCCCNC(=O)CC1CC1 C1(CC)(NC(=O)CCc2nc[nH]n2)CCN(C(=O)CCn2ccccc2=O)CC1 c1(C(=O)NCc2cccc(NC(C(C)(Cl)Cl)=O)c2)c(F)ccc2ccoc12 N1(C(CSCC(N)=O)=O)CCC2(NC(c3nc(C4CC4)cs3)=O)CC2C1 C1(NC(C2(C(C)C)CCC2)=O)COC2C(NC(=O)C(C)CC(C)(F)F)COC12 CC1CCN(C(=O)CC2CC(F)(F)C2)CCN1C(c1cc(C(N)=O)cn1C)=O C(=O)(CC(CC(C)C)NC(=O)CC1CCC(=O)CC1)N1CC(CCCCC)C1.CC C=CCC(C(=O)NCCCC(O)CO)NC(=O)CC(C)SC C(CCN=c1[nH]cc([N+](=O)[O-])cc1CO)N(C(c1cc(C)nnc1O)=O)CCO Cc1n[nH]c(=NC2(C(N)=O)CCN(C(c3cnsc3C)=O)CC2)o1 c1(C(N2CC(CC)N(C(c3ccc(C)o3)=O)CC2)=O)ccn2c(C)cc(C)nc12 C(=O)(CCCCNC(=O)CCC(=O)NC1CCCC1)N(CC)CC1CC1 n1(CC)cnc2c(NCC(C)(C3CC3)NC(=O)C=Cc3ccc(C)o3)ncnc12 c1(OC)ccc(C(N2CC3CN(Cc4ccc(F)cc4Br)C3C2)=O)c(OC)n1 c1(OC)cc(C(N2CCCC(CCCCNC(c3ccno3)=O)C2)=O)ncn1 Cc1cc(O)cc(=O)n1CC(=O)NC1(CN(C(=O)C(O)CN2CCCC2)C)CC1 c1(C(N2CC3N(C(c4c(F)ccc(C)c4)=O)C3C2)=O)cc(O)c(O)c(O)c1 CCC(C#N)C(=O)NCC1CC(COC)CN1C(=O)CCCc1cc(C)sc1C c1(C(N(CCN(C(=O)CCN(S(C)(=O)=O)C)C(C)C)C)=O)cnc(C2CC2)o1 C1(CC(=O)N(C2CN(CC(F)(F)F)C2)C)CCC1(C)C C1(NC(CC(C=C)(C)O)=O)C2CC(O)C1N(C(=O)C(c1ccc(Cl)nc1)(C)C)C2 c1(OCC)ccc(C(=O)N(CC(CC)NC(=O)C2=COCC2)C)cc1OCC c1(CC(=O)NCCCNC(C(=Cc2ccccn2)C)=O)ccc([N+](=O)[O-])cc1 c1(C(=O)NC(CNC(C(CSC)OC)=O)C2CC2)cc(O)nc2cnccc12 CC1CCC(O)C(NC(C2(CNC(c3csc(=N)[nH]3)=O)CCCO2)=O)C1 n1(CCCCC)cc(CNC(C2CC(NC(=O)OC(C)(C)C)C2)=O)c(C)n1 c1(N2CCc3c(ccc(OC)c3)C2)nc(=NCCCNC(C)C)[nH]c2ccsc12 c1(C2(C(N(CC(CN(C)C(c3cccs3)=O)O)C)=O)CC2)ccccc1Cl c1(C(=O)NCC(C2CCOC2)NC(C2(OC(C)=O)CC2)=O)cc(S(C)(=O)=O)cs1 Cc1nncc(C(N2CC(C)(NC(C3COCC(C)O3)=O)C2)=O)c1C C=CCCCC(C(=O)NC1CC1C1CCCCC1)NC(c1cnc(C)s1)=O N1(C(c2cccc(CC)c2O)=O)CC(C)N(C(=O)CCc2nccs2)C(C)C1 C=C(C)CCCC(=O)NC1CCCN(C(=O)C(C)CC2CCCC2)C1 N1(C(CC2(OC)CN(C(c3c(CC)ocn3)=O)C2)=O)CCN(C)C2CC12 C1(CNC(CCC=C(C)C)=O)COC(C)(C)CN1C(=O)C=Cc1ccc(F)cc1 CC(C)(C)C(CNC(c1cccnc1F)=O)NC(c1cccnc1Cl)=O C12(CC(=O)NC(C3CCN(C(c4cscc4Cl)=O)CC3)C)CCCCC1C2(F)F C(=O)(CC(C)(O)C(F)(F)F)N1CC(NC(c2c(C)noc2)=O)C1 N1(C(c2c(C)ncc(C)c2)=O)CC2CCC1CN2C(=O)Cc1cc[nH]c(=N)c1 CC(CC(=O)NCC1CN(C(=O)CNC(C2CCC2)=O)C1)CC(C)(C)C c1(N(C)CC2CCCCN2C(C2COC3COCC23)=O)nc2cccnc2s1 N1(C(CC(=C)I)=O)CCC(CO)(CNC(C2(CO)CC2)=O)CC1 CC(C(=O)N1CCOC(CN(C)C(c2ccccc2C2(C)CC2)=O)C1)S(C)(=O)=O C1(CCNC(C=C(C)C(F)F)=O)CCN(C(C2(C)CCCCO2)=O)CCC1(F)F C(=O)(C1=C(C)OCCC1)NC1CC2(C(C(N(C(CC)CC)CC(C)C)=O)C2)C1 c1(C(=O)NCC2(CNC(c3csc(Br)c3)=O)CC2)cncc2[nH]ccc12 CC#CCC(C(=O)N1CCOCC(O)C1)NC(c1occc1CC)=O N1(CCC)C(=O)CCC1C(=O)NC1(C2CCCN2C(=O)CC2CSCCO2)CC1 CC(C)C(CN(C)C)C(=O)NC(CNC(=O)C=C1CCC(C)CC1)C(C)(C)C CC(C)(O)C#CC(=O)NCC1CC(C(=O)NCc2ccncn2)CO1 C12(CC(=O)NCC3C(NC(CC4CCC(C)(C)CO4)=O)C3)CCC(CC1)C2(C)C Cc1ccc(C(=O)NCC2=CCN(C(C3CCSC3)=O)CC2)nc1O c1(CCNCC(=O)N(C)CCc2ccccc2)ccc(Br)cc1 c1(C(=O)NCC(CC)NC(C(C(C)C)SCC)=O)cccc2c1CC(=O)N2 C1(C2CCOCC2)(C(=O)NC(C(=O)O)c2cscn2)CCNC1 C(C(C(C)C(C)C)NC(=O)CSCC(C)C)NC(COc1cccc(C)c1)=O C(S(=O)(=O)c1ccc(-n2cc(C)cn2)cc1)c1onc(-c2scc(C)c2)n1 Cc1cnc2c(C(=O)NCC3CCN(C(C4CC(CN(C)C)C4)=O)C3)cnn2c1 CC(C)C(C(=O)NCCC1(O)CCN(C(c2cscc2F)=O)C1)NC(N)=O N1(C(CCOCC#C)=O)CCN(C(=O)CNC(=O)C(C)(C)c2ccc(Cl)s2)CC1 CCCS(=O)(=O)C(C)C(=O)NCCC1CC2CCC(C1)N2C(=O)CCCC(C)=O c1(C(=O)NC2CN(C(C(C)(C)C3CCCC3)=O)CC2F)ccc(F)c(C(F)F)n1 c1(OC)cccc(F)c1C(=O)N(CC(C)CNC(=O)CC1CCCN1C(C)C)C CC(C(=O)N(CCCN(C(=O)C(C1CCCO1)C1CC1)C)C)OCCN(C)C C(=O)(CCC(F)(F)Cn1cc(C2CCCCC2O)nn1)N1CC(S(C)(=O)=O)C1 C1(C(=O)NC(CCCN(C(CN(C(=O)OCC)C)=O)C)C)CC(CC)C(OC)C1 CC1(C)C2CCC1(C)C2C(=O)NC1CN(C(C2CCC(C(N)=O)O2)=O)CC1C1CC1 S(=O)(=O)(c1cc(C)cnc1NCCCSC)N1CCCC(C)(CCC)C1 N1(C(c2c(COC)cccc2)=O)CCN(C(=O)CCCCNC(N)=O)CC1CO C(=O)(C(C)(C(C)(C)O)NCC1CNCCN1C)OC Cc1nc(NC(C)(C)CNC(=O)CC2CC2(C)C)c2c3c(sc2n1)CCC3 CN1CCC(C)(CNC(=O)CC2(CNC(=O)C(C)(C)F)CC2)C1 C1(C(=O)NC2C(N(C(=O)CC(F)(F)F)C)CCCC2)Cc2cc(Br)ccc2O1 C(CN=c1[nH]c2c(C(F)(F)F)cccc2c(=O)n1C)c1c(OC)cc(OC)nc1 N1(C(C(C)C2CCC2)=O)CC2(C)CN(C(=O)CCC3CC3(Cl)Cl)CC2(C)C1 C1(C(=O)NC(C(C(=O)N(C2CCCC2)CCOC)C)C)CC12CCCCC2 c1(OC)cc(C(=O)NCC2C3CC2N(C(=O)CN2CCC(C)C2)C3)ccn1 c1(C(N2CCN(C)C(=O)C2)=O)cc2ccc(C3=COCC3)cc2o1 c1(CCN(C(CC2CCC2)C(=O)NCCOC2CC2)C)ccccc1 c1(C(=O)NCC2(OC)CN(C(CCC#C)=O)C2)c(OC)ccc2c1CCC2 c1(C(=O)NC(C)CNC(=O)COC(C)(C)C)c(-c2ccccc2)noc1C1CC1 N1(CC(c2ccc(-c3nn[nH]n3)cc2)C)CCCC1(C)Cc1ccsc1 C(=O)(C1=NN(CCO)C(=O)CC1)NC(C1CN(C(C2(C)CCC(=O)N2)=O)C1)C CS(=O)(=O)c1ccc(C(=O)NCC2CCC2NC(c2ccc3nsnc3c2)=O)[nH]1 Cc1cc(CN2CC(O)CC2C(N2CC3CCC(C2)O3)=O)cc(O)c1 N1(C(Cc2c(C)cc(C)s2)=O)CC2(CCN(C(C3CCCN3C3CC3)=O)CC2)C1 c1(CC)cc(C(N2CCCC2CN(C(=O)CC2(C)CC2(F)F)C)=O)no1 C1(OC)CCCCC1C(=O)N(C(C)CNC(=O)CSc1cccs1)C Cc1ncsc1C=CC(=O)NCC1CC1NC(=O)CCCc1ccccn1 C1(C(NOCCC(=C)C)=O)(CC)CCCN1C(C1CCC(C2CC2)CC1)=O CCCCCC(C)CC(=O)N1CC=CC(NC(C2CCCN2CC)=O)C1 C(CCCC(C)NC(C12CC(F)(C1)C2)=O)NC(c1n(CC)ncc1)=O CCC(C(=O)NCC1CCN1C(=O)C(C)(C)c1ccccn1)NC(N)=O c1(C(=O)NCC(C)(C)OCC(=O)Nc2cnc(CO)s2)cccc2cncn12 C1(C(=O)NC2(CC)CCCC2)CN(C(C2CCC=CCCC2)=O)CC1(F)F c1(C(N2CC3C(CC(=O)NC(c4nccs4)C)C3C2)=O)cnn2cccnc12 C12(CC(=O)N(C)Cc3nnc(O)o3)CCC1CN(C(c1csc(CO)n1)=O)C2 C(=O)(C=C1SCC(=O)N1C)NC1CN(C(CC(C)C(F)F)=O)CC1(C)C C(CC)(C(F)(F)F)C(N(C(CO)C=O)C)=O.c1(C(C)=O)cnn(C)c1 C(=O)(C(O)C(C)(C)C)NC1(CC(=O)NC(C2CSC2)C)CCCCC1 N1(C(CC23C(CN(C(c4cnn(C)c(=O)c4)=O)C2)CC3)=O)CC2(C)CCC2(C)C1 C1(C2CC2)(CNC(C2CCN(C)CC2)=O)CCN(C(=O)C(C#N)=CC2CC2)C1 c1(OC)cc(C(=O)NCC2CC(NC(=O)C(C)CC(F)F)C2)c(Cl)cn1 C#Cc1ccccc1CC(=O)NCC1CCN(C(c2ocnc2C2CC2)=O)CC1 c1(C(N2CCC(CCOC)(NC(C(C)OCC#C)=O)C2)=O)c(OC)ccnc1O C#Cc1cccc(C(=O)NCC(F)CNC(=O)C(C)n2ccnc2)c1C c1(C(N2C(COC)CN(C(=O)CC(C)C(F)F)CC2)=O)cc(O)cc(N)c1C C(CCOC)(C(N)=O)NC(CCN(CC#C)C(c1cc(C)cs1)=O)=O CCC(C)(C#N)C(=O)NCC1(C)CCCN(C(c2ccc(Cl)cc2)=O)C1 C(=O)(C1=CCC2CCC1N2C(=O)CN1CCCC1=O)NC1CC(C)n2c1ncc2 N1(C(C2C(C)CCC2)=O)CC2=C(C1)CN(C(c1ccc(O)c(Br)c1)=O)C2 CC12OCC(NC(c3cccn4cnnc34)=O)(CO1)CO2 CC1=C(C(=O)N2CCCC2CN(C(=O)CNC(c2ccc(C)s2)=O)C)CCCO1 N1(C(c2snc(C)c2N)=O)CCOCC(C(=O)N(C)CC2C(C)(C)C2(C)C)C1 C1(CCC)(NC(=O)CCN(C)CC)CCCN(C(=O)CCC2CCCC(=O)N2)C1 Cc1cc(C(=O)NC2CN(C(=O)CCC3CCCCCC3)CC2C)c(C)o1 N1(C(CCCNC(C2(COC)CCCC2)=O)=O)CCCC(O)(CO)C1 CC(S(=O)CC(=O)N1CCCCC1)c1nccc(O)n1 CN=C(NC(=O)C(C)Cc1ccncc1)N(C)CC1(CO)CCC1 N1(C(CCOCC#C)=O)CCN(C(C2CC2(C)C)=O)C(CC)C1 N1(C(CCC(C(C)C)NC(c2cc(Cl)no2)=O)=O)CCC2(CC1)CC(O)C2 CCCCC(CNC(C1(CO)CCCO1)=O)NC(C12CCC(CC1)C2)=O N1(C(CC(CN(C)C)O)=O)CCCC(CO)(NC(=O)CSC(C)(C)C)C1 c1(OC)c(C)cc(C(=O)NCCNC(=O)C=CC(c2ccc(C)cc2)=O)cc1Cl C(=O)(C(N)CCC(N)=O)N(C1CC2CNC1C2)CCN1C(C)(C)CC1 CCCCS(=O)(=O)NCC(=O)NC(C)(CNC(C1CCCC1)=O)C1CCC1 c1(-c2cn(CC(=O)NCC3C(C)C3C)nn2)ccc(C(=O)O)c(F)c1Cl c1(OC(C)C)cccc(C=CC(=O)NC(C)CCNC(=O)C=CC(=O)N(C)C)c1 c1(CC(=O)NCCN2CCCN(C(C3C(C=C)C3)=O)CC2)csc2ccccc12 N1(C(c2cc(OC)n[nH]2)=O)CCN(C(=O)COCCc2cccs2)C2CCCC12 C(C(C)(C)C(C)(C)O)NC(C(CC)N(C)C(c1nccs1)=O)=O c1(NC(N)=O)ccc(C(N2CC(NC(C3CCCC34CC4)=O)C(O)C2)=O)cc1 Cc1ccc(C(N2CCC(OCC(=O)NCC3(F)CCN(C)C3)C2)=O)nc1C c1(SCC(=O)NCC2CCN(C(C3CCC(CC)O3)=O)C2)cccc(C(C)C)c1 C(=O)(CCC(F)(F)CCOC(c1cnn(-c2ccccc2)n1)=O)OCC N1(C(c2nc(OC)c(F)cn2)=O)CCC2(CCC2NC(=O)CC(C)(C)C)CC1 Cc1cc(C2CCC2)ccc1C(=O)NCCNC(=O)CCCN(C)C(C)C N1(C(c2cccc(C)c2N)=O)Cc2[nH]nc(C(=O)NC3CCN(C(C)C)C3)c2C1 C(=O)(C1(C)NCCc2ccsc21)Nc1cc(C(=O)OC)cc(C(F)F)c1 C(=O)(CC(C)CC(C)C)N1CCN(C(c2ccc(CC)s2)=O)C(CC(=O)NC)C1 N1(C(CCC2C(C)(C)C2)=O)CCCC12CCN(C(=O)CNC(N)=O)CC2 N1(C(c2oc(C)c(-c3ccccc3)c2)=O)CCOCC(CNC(=O)CC(C)(C)O)C1 C(=O)(C1=CCOCC1)NC1CCN(C(CCC(=C)C)=O)CC1.N12CCC(CC1)C2 C(C)(CCNC(C1(C)CC1C(F)(F)F)=O)NC(C=CCOC)=O N1(C(C)=O)CCC(C)(C(=O)NCC2(O)CCCN(C(=O)COC(C)C)C2)CC1 n1(C2CCCN(CC(CCOC)O)C2)cnc2ccccc12 C(N=c1[nH]c2c(c(=NCC3CCC4CC34)[nH]1)CCCC2)c1ccc([N+](=O)[O-])cc1 N1(C(C(C)NC(C)(C)C)=O)CC2CCC(NC(=O)C=CC3CCCC3)(C2)C1 c1(C(=O)NC(C(=O)OCC)C)csc(N=S(C)(=O)c2cccc(OC)c2)n1 C#CCC(C)(C(=O)NCc1cccc(C)c1C)NC(=O)C=C(CCC)CCC c1(C(=O)NCC2C(NC(=O)CN3CC4CC4C3)C2)cc2ccncc2[nH]1 C1(NC(C(CSC)C)=O)CCN(C(c2sncc2C)=O)C12CCC2 C12(NC(Cc3cccc(CC)c3)=O)CCN(C(=O)CC3CCOCC3)CC1C2 CN1CCCC(C(=O)NC2C=CC(C(N3C(CO)CC3CO)=O)C2)C1 Cc1cc(C(N2CCC(NC(C3(C)C=CCCC3)=O)C2)=O)ncc1CO c1(C(C(=O)NC2(C)CC2)N(C(CCCC)C)C)ccc2ncsc2c1 N1(C(c2ccc(OC)cc2O)=O)CC2CC1CN(C(C1CC1C(C)C)=O)C2 c1(C(=O)NCC(CC(C)C)NC(=O)CC(C)N(C)C)cc(S(N)(=O)=O)ccc1O CC1CCCC(c2nnnn2C)(NCC2=CCCCC2)CC1 C1(c2n(CCNC3(CCF)CCC3)nnn2)(OCC)CC2CCCC(C2)C1 c1(CC(=O)NC2CN(C(C(CC)CC)=O)C(C)C2)[nH]c(C(C)=O)c(C)c1C(=O)OC CC1(C)CCN(C(C2CC2(Cl)Cl)=O)CC1NC(c1coc(C2CCCCC2)n1)=O C(N=c1[nH]c(Cl)nc2[nH]ccc12)C1CCC(NC(C2C(CC)OCC2)=O)C1 C12(OC)CCC(C(=O)NC3CC4CN(c5cc(Cl)nc(C(C)C)n5)CC34)(CC1)C2 c1(NC(C(=O)Nc2cn(CCOC)nc2)=O)cc(Br)cnc1N(C)C C=C(Cl)CCC(=O)NCC1(C)CCC(NC(c2nc(O)c(C)s2)=O)C1 Cc1cc(Br)cc(S(=O)(=O)N2CCCC(C)(C(=O)Nc3ccc(Br)cc3O)C2)c1 c1(OC)ccc(C(N)=O)cc1C(=O)NC1CC(CNC(c2cc(Cl)n(C)n2)=O)C1 Cc1ccn(C)c(=O)c1NC(=O)C(Cn1cncn1)NC(C1CCCN1C)=O C(=O)(C(Cc1ccccc1)C(F)(F)F)N1CC(C)(NC(C2(F)CCOC2)=O)C1 C12(NC(C(C)=C3CC3)=O)CC3CC(C1)CC(NC(C1CCCC(O)C1)=O)(C3)C2 C(=O)(C1Cc2ccccc21)NC1C(C)(CNC(C2CC(CC)(CC)C2)=O)CCC1 CC1(C)CC(C(N2CCCC2C(=O)NCCCCC2CC2)=O)CCO1 CN1CCC(CN=C(NC2CC2)NC2CCN(C(=O)CSC3CC3)C2)CC1=O c1(C(=O)NCC(COC)NC(=O)CC2CCCN2C(C)=O)cccc(C)c1F C12(C(=O)NCC(CNC(C3CC4CC4C3)=O)CO)CCC(CO)(CC1)C2 N1(C(CCC2(OC)CN(C(=O)C3=CCCOC3)C2)=O)CC(C)OC(C)C1 CC1(C)CC(C(=O)NCC2CC2NC(=O)C=C2CCSCC2)C1 c1(CC)cc(C(=O)N(C)CCN(C(c2cnc(C3CCOC3)s2)=O)CC)ncn1 C1(NC(CSCCCC)=O)CN(C(C2(F)CCCCC2)=O)CC12CCS(=O)(=O)CC2 N1(CC)CCOCC1C(=O)NCCCCNC(=O)C(C)C1CCCC1 Cc1c(CC(=O)NC2CC2NC(C2CCC(C(N)=O)C2)=O)ncn1C CC(CC(C)(C)C)C(F)C(=O)NCCCCCN(C)C(c1cc(C2CC2)on1)=O c1(OCC)ccccc1N(C(c1cc(C(C)(C)C)on1)C(=O)NCC1CC1)C C1(C(=O)Nc2cncc(C(F)(F)F)c2)CN(C(c2ccccc2Br)=O)CCC1O C(=O)(CCC(=O)C1CC1)NCC1CCC(NC(CSCCC(C)C)=O)C1 c1(OCC=C)ccc(C(=O)N(C2CN(C(=O)CC(C)n3cccn3)C2)C)cc1 N1(C(c2cc(C(F)(F)F)nn2C)C(=O)OC(C(=O)NC)C)CCCCC1C c1(OC)cc(NC(c2nc(CC3CC3)no2)C)[nH]c(=N)n1 N1(C(c2c(C)ccnc2C)=O)C2CCC1CN(C(c1nccc(Cl)c1O)=O)C2 CCCCCCC(C(=O)N1CCOC(CNC(=O)Cc2ccco2)C1)NC(C)=O CCCC(C)(CO)NC(C1OCCC1NC(=O)CC(C)O)=O C12(C(=O)NCCCN(C)C(C3CC34CC4)=O)CCCC(CCC1)C2O CCCC(C(O)C(=O)NCCC1CCCC1)NC(C1CCC2(CC2)C1)=O c1(C(N(C)C)=O)cccc(Cl)c1N(C(c1ccc(F)cc1)=O)CC1CCC1 C(C(C)NC(=O)CSCc1c(C)noc1C)(C(C)C)NC(c1cc(C)ns1)=O N1(C(c2cnc(CCC)s2)=O)CC(NC(=O)C(C(C)(C)C)C2CCC2)C2(CC2)C1 Cc1ccc(O)cc1C(=O)NC12CC(C(N3CC4C(C3)C4(F)F)=O)(C1)C2 CC1CN(C(=O)C(C)N(C)C)CC1NC(c1ccc(-c2ccccc2)s1)=O c1(OCCC)ccc(C(=O)NCCCCN(C)C(C2(C)CCN(C)C2)=O)cc1 c1(C(N(CC(CC)NC(C2CCC(=O)O2)=O)C)=O)oc2ccc(OC)cc2c1C n1(CC(=O)NC2CC(NC(=O)CNc3ncccn3)C2)cccnc1=O CCCCCC(O)CC(=O)NC1CCN(C(c2ccn3cccc3c2)=O)C1(C)C C1(C)(NC(CC2(C)N(C(Cc3n(C)cnc3)=O)CC2)=O)CC(C)(C)OC1=O c1(C(C(OC)OC)NC(=O)Cc2ccccc2)ccc(C)cc1 C1(C(=O)NC(CNC(c2cnc(CC)[nH]2)=O)C2CCC2)CC2(C1)CC2F c1(CNC(C2N(C(C(C)CC3CC3)=O)CCC2O)=O)cnc2n1CCC2 C1(C(=O)OCCC(=O)N2CCCC2)CCCCC1N1CCOCC1 N1(C(C(C)C2(O)CCC2)=O)CCC2(CC2)CC1C(=O)NC1CC1 c1(C(=O)NC2CCN(C(c3c(C)cc(C)nc3)=O)CC2O)ccc2nn[nH]c2c1 c1(C(N2CC(O)(C(C)NC(c3cn4ccsc4n3)=O)C2)=O)[nH]cc2c1CCCC2 C1(C)(C(=O)OC)CCN(C(C2CN(C(=O)CC(C)N(C)C)CC2N(C)C)=O)C1 c1(C(N2C(CCNC(=O)CCC3CCC3)CC(OC)C2)=O)cccc(C)c1Cl N1(C(C2C(=C)CC2)=O)CCN(CC(C)NC(c2c(C)nsc2Br)=O)CC1 N1(C(C(CC)COC)=O)CCC(O)C(NC(C2(COC)CC2)=O)C1 c1(C(=O)N(C)C)cccc(C(=O)NCC(CC)NC(C23CCC(OC)C2C3)=O)c1 N1(C(c2nc(COC)oc2)=O)CCC2C(NC(C34CC(F)(C3)C4)=O)C2C1 c1(C(N2C(CN(C(=O)C3=C(Cl)CCCC3)C)CCC2)=O)cc2ccncc2s1 c1(CNC(CCSCC)=O)ccc2c(c1)CCCC2NC(=O)C=C1CCCCC1 C(=O)(C(CNC(c1cc[nH]n1)=O)C(C)(C)C)N(CCN1CC=CC1)CC Cc1nc(CCNC(=O)C(CN(C)C)NC(=O)CC(C)n2cccn2)n[nH]1 c1(SCCC)nc(Cl)c(N)c(=NCCc2nnc3n2CCOC3)[nH]1 c1(C(=O)NC2(CCNC(=O)C=CC3CCOC3)CC2)cc(O)cc(F)c1 c1(C(=O)NCCCC2N(C(=O)COCCOCCF)CCC2)ccc(OC)cc1 c1(C(=O)NCC2(C)CCN(C(=O)CC3CCNC3=O)C2)cc(O)nc(O)c1 CCCC(C)(C)C(=O)NCCOCCN(C)C(C1(CO)CCC1)=O C12(NC(CNC(=O)NC)=O)CCC(CNC(=O)C(C(C)O)N(C)C)(C1)OC2 C1(NC(Cc2cnn(C)c2C(F)F)=O)COCCN(C(C2CC(=O)CO2)=O)C1 n1(CC)nc(C)c([N+](=O)[O-])c1NCC1CN(C(=O)C2=CCCCC2)CCC1C N1(C(c2c(C)nn[nH]2)=O)CCOC2(C1)CN(C(=O)C(C)C(C)C1CCCCC1)C2 N1(C(CC(COC)NC(c2sccc2CO)=O)=O)CCC(N=[N+]=[N-])C1 c1(CCC(=O)NC2CC(NC(=O)CC34COCC(C3)C4)C2)ccccc1Cl C1(NC(c2cccc(NC(=O)OCC)c2)=O)CN(C(=O)C#CC2CC2)CC12CC2 c1(C(N(CCN(C(CC=C=C)=O)C)C(C)C)=O)cnn(CC(F)F)c1C C#CC1(C(=O)NC2CC23CC(OCC)C3)CN(C(=O)CC(C)O)C1 c1(NC(=O)NCC(CCC)C(=O)OC)cc(C)cc(Br)c1F c1(C(=O)NCC2CC(NC(COCC(C)C)=O)C2(C)C)ccc2sccc2c1 N1(C(C(C)N(C)C)=O)CCN(C(c2cn(CCO)nn2)=O)C(CC(F)(F)F)C1 O=C(CC1CCc2ccccc21)N1CC(C2CN(C(=O)C(O)C3CCC3)C2)C1 CC1CCCC(C#N)(NC(C2CCCN(c3ccccc3)C2)=O)C1 Cc1ccc(NC(N2C(C(=O)NC(C)C(F)(F)F)CCC2C)=O)cc1 C1(CCC)CN(C(=O)C(CCO)N(C)C)CCN1C(=O)CC1(O)CCCCC1 C(=O)(C1=Cc2cc(F)ccc2OC1)NCC(C)NC(C1CC(C)(F)C1)=O c1(C(=O)NCC2CC(F)(CNC(CCC=CC)=O)C2)ccc(N(C)CC)cc1 c1(C(N2CC(C(c3cn4ccc(Br)cc4n3)=O)C2)=O)c(Cl)[nH]c2ccccc12 c1(CNC(C2CN(C(N)=O)C2)=O)ccc(C(N2CCC(CCO)C2)=O)o1 c1(C(=O)OCC)cc(NC(=O)Nc2cccc(NCCN=[N+]=[N-])c2)ccn1 C1(C)(C(N(CCCNC(C(C)n2cncn2)=O)C)=O)COC(=O)C1 CC1(C#CC(=O)N2CCCCC2C(N2CCSC3(CCC3)C2)=O)CCCO1 C1(NC(COCC)=O)CCSC12CN(C(=O)CC1CCCC3(CC3)C1)C2 C(=O)(C(F)CCC(C)C)N1CC(C(C(=O)NCC2(C)CCC(=O)N2)OC)C1 C=C(C)CC(C(=O)NCc1cccc(CC2(NC(=O)CC3CSC3)CCC2)c1)OC CC1CN(C(c2cc(C(N)=O)cn2C)=O)CCCN1C(=O)CC1=NNC(=O)C1 C1(C(=O)NCC(CN(C(C(C)O)=O)C)O)CCC2(CCC2)CC1 N1(C(CC#N)=O)CCCC1C1(C(=O)NCc2cscc2C(F)(F)F)CC1 c1(NC(c2csc(C3CC3)n2)=O)ccc2c(n1)CCCC2=O CCCCCCC(C)C(=O)NC1CCC(NC(c2cc(C#N)c(C)cn2)=O)C1 Cc1ccc(C(=O)NC2CC3CC2N(C(c2cccc[n+]2[O-])=O)C3)cc1C1CC1 c1(C(=O)OCC)n[nH]c(=NC(=O)OC2CCCC(C(=O)N(C)C)C2)s1 N(C(=NCCCOC(=N)O)NCC(C)(F)F)CC(C)C1CCC1 Cc1ccc(N)c(C(=O)NC(CO)C(C)NC(c2cn(C3CC3)cn2)=O)c1F N1(C(C(C)=CC2CC2)=O)CCCCC(NC(c2cnc(C(F)F)cn2)=O)C1 CC1CC(CNC(c2ccsc2Cl)=O)CN1C(=O)COC1CCCCC1 c1(CNc2c(C(=O)Nc3c(I)ccc(C)c3)ccc(Cl)n2)cc(F)c(C)c(F)c1 Cc1[nH]nc(C(F)(F)F)c1C(=O)NC(C)CNC(C1(C)CCC(=O)N1)=O c1(CC(=O)NCCN(C(C(CC=C)CC)=O)CC)noc2ccccc12 CC(C)(F)C(C)(F)C(=O)N1CC2(CC(NC(=O)Cc3cncc(C#N)c3)C2)C1 C(C(C(=O)N1CCCC(C(C)C#N)C1)C(C)C)NC(c1c(C)[nH]nc1CO)=O N1(C(C2(CC)CN(C(c3cscc3OC)=O)C2)=O)CC(C)=CC(C)C1 N1(C(CC=CCC)=O)CCC(C2(O)CN(C(=O)Cc3ccc(C#N)nc3)C2)CC1 CC1CCN(C(c2ccco2)=O)CC1NC(C12CCC(C(F)(F)F)(CC1)C2)=O c1(C(C)NC(c2cnc(Cl)s2)C)cncc(Cl)c1 c1(C(N(C(C)CNC(=O)C=C2CCCCC2)C)=O)cc(Cl)ccc1O c1(CC(=O)NCC(C)N(C)C(C2CC(N(C)C)C2)=O)ccc2c[nH]nc2c1 C1(CNC(C2(CC#C)CC2)=O)(COC)CCN(C(=O)C(C)CO)C1 N1(C(COCC)=O)CCN(C(=O)Cc2ccc(C)c(O)c2)C(C2CCC2)C1 c1(C(C)=O)cc(Br)ccc1NC(=O)NCC1OCC1(C)C n1(CC(=O)NC(C)COC(C)(C)C)cc(CCC2CCCCC2)nn1 N1(C(CCNC(N)=O)=O)CCC(CO)(CNC(=O)CSC2CCCO2)CC1 c1(-c2ccccc2)cccc(N2CCN(CCC3CNC3)CC2)c1 C1(C(N2CCC(C(=O)NC(C3COCCN3C)=O)C2)=O)CC2CC2N1CC O=C(CC1=CCN(C(=O)C(F)C2CCC2)CC1)NCCCc1ccncc1 c1(CN2CC(C(=O)Nc3ccns3)C(O)CC2)cccn2ccnc12 CC1CN(C(c2cc(C3CC3)no2)=O)CCC12CCN(C(=O)C(C)C1CC1)CC2 c1(NC(C2COc3ccccc3C2)CSC)ncc(F)c(=NC2CCCCC2)[nH]1 N1(C(=O)OC(C)(C)C)CC(C(N2CCCCC(C)(F)C2)=O)CCC12CC2 N1(C(C(CC)O)=O)CCN(Cc2c(Br)c(C(F)(F)F)nn2C)CC1COC c1(C(C(=O)NCCCF)N(CCC)CCN(C)C)cccc(C(=O)OC)c1 c1(CC(C(=O)NCCC(F)F)NC(C2CCCC3CC23)=O)ccccc1Br C1(NC(=O)Nc2cn(C3CCOCC3)nn2)CCN(C2CCCCC2)C1=O N1(C(c2cc(C)on2)=O)CCC(CCCCNC(C2CCOCC2)=O)CC1 C1(C(=O)NCCOC(C(C)N(CC)CC)=O)CC1(C)CC CC1Cc2sc(C(=O)Nc3ccsc3COC(C)C)cc2C(C)C1 CCC(O)C(C)C(=O)NC(C1CN(C(C2CCN2C)=O)C1)Cc1ccccc1 C(=O)(CC(=O)N1CCCC1CN(C)C(c1cc(CC)[nH]n1)=O)OCC N1(C(CNC(C)=O)=O)CCOC2(CCS(=O)(=NC(=O)c3cc(C)ccn3)CC2)C1 Cc1sncc1C(=O)NC1(C(=O)N(C)CCC2CCCO2)CC(F)C1 N1(C(CNC(=O)OC)=O)CC(NC(=O)Cc2ccccc2C(C)C)C(C)C1 N1(C(C2(SC)CN(C(=O)C(C)C(F)F)C2)=O)CC(CO)C2(CC2)C1 c1(N2CCCC(C)(C)CC2)nccc(=NCCCNC(=O)C2CC2)[nH]1 C(=O)(CCCC(C)=O)NCc1cc(C(=O)NCCCCC)n(C)n1 C1(C(N2C(CC)CC(C)C2)=O)CCC2CCC1N2C(=O)CCC1CCCN1C C1(NC(c2ccc3c(c2)OCC3)=O)CN(C(=O)Cc2cscn2)C2(CCOC2)C1 C(=O)(CCCCCC(C)C)NCC(C(=O)N(CC)CC1CC1)N(C)C C1(NC(C=C(C)C)=O)CN(C(c2ncncc2Cl)=O)Cc2ccnn2C1 C12(C(=O)NC(c3cncnc3)C)CC1CN(C(c1nocc1Cl)=O)C2 Cc1cc(C(N2CCC(NC(=O)C(C)C)C(O)C2)=O)c2c(C3CC3)noc2n1 C1(CC=C)(NC(=O)CC(C)SC)CCN(C(=O)C(C)C#N)C1 C1(OC)CN(C(c2cccc(O)c2)=O)CC1C(=O)NCc1ccncn1 c1(SCC(=O)N2CCC2CNC(C2(O)CCCCCC2)=O)cc(Cl)ccc1Cl c1(C(N2CCN(C(C(C=C)O)=O)CC2CC)=O)cc(S(=O)(=O)NC(C)C)c[nH]1 c1(C(N(CCCN(C)C(c2cc[n+]([O-])cc2)=O)C)=O)[nH]nc2c(=O)n(C)cnc12 c1(C(=O)OC)occc1C(=O)NCCOCCOCCNC(=O)C(CF)CF c1(C(N2CC(C(=O)NC3COCC3O)C2)=O)cc(F)ccc1C(F)(F)F CCC(C(=O)NCC1CN(C(C2(C(C)(C)C)CCC2)=O)C1)C(C)C c1(CC)onc(C(=O)NC(C)(C)C(C)NC(C2CCN(CC3CC3)CC2)=O)c1C CCCCCC(O)C(=O)NCC1CCN(C(c2ccc(CC(C)(C)O)s2)=O)C1 N1(C(CC2(OC)CC2)=O)C2CCC1CN(C(=O)C(C)Sc1ccccc1C)C2 C(=O)(C(CC(=O)NC(CNC(c1cc(Cl)cc(Cl)c1)=O)C(C)C)C(C)=O)OCC Cc1c(C(=O)NC(CNC(C23CC(C)(CO2)C3)=O)C(C)(C)C)cnc2nncn12 n1(C(C(=O)NC2C(CC)CN(C(=O)C=C3CCC3)CC2)C)cc([N+](=O)[O-])nc1C c1(C(C(=O)NC)N(C)CC2CCCN(C)C2=O)ccc(Br)c(C(F)(F)F)c1 c1(C(N2CC(CNC(c3c(COC)scc3)=O)OCC2)=O)cccc2oncc12 Cc1oc2ccccc2c1C(=O)NC1CN(C(C2CC(S(C)(=O)=O)C2)=O)C2CC12 C1(C(=O)NCCCN(C)C(c2cnnn2C)=O)CCC12CCCO2 N1(C(c2c(C)ncs2)=O)CCN(C(C2(C)CCCO2)=O)CC1c1ccccc1Cl C1(C(N2CCCC(CCNC(C=CCCC=C(C)C)=O)C2)=O)CC2(CC(=O)C2)C1 C1(CC)CCCCC1N(C(=O)C(=O)NCCOC1(C)CCOCC1)C C(=O)(C(C)C(F)(F)C(F)F)N(C1CCCN(C(c2c(C)cnn2C)=O)C1)CCO CC1=CCC(C(=O)NCC23CC2CN(C(c2ccc(C(C)(F)F)nc2)=O)C3)CC1 C(C)(CCC(=O)Nc1cc(C)sc1C)NC(c1ccc(SC)o1)=O c1(C(N2CC(O)CC(NC(c3c(C)csc3)=O)C2)=O)cccc2c1C(=O)NC2 C(C=CS(F)(F)(F)(F)F)N(C1CCC(c2ccccc2)CC1)C C1(NC(C2=CC(C)(CC)C2)=O)CCCCN(C(c2n[nH]c3c2CCC3)=O)CC1 c1(C(C(=O)NCCCSC)N(C)CC2(O)CCOC2)n[nH]cc1Br N1(C(CCn2c(C)nc([N+](=O)[O-])c2)=O)CCN(C)c2ccc(Cl)cc21 C(=O)(C(C)=Cn1ccnn1)N1CC(CCNC(CC2(COC)CCOCC2)=O)C1 N1(C(C(c2ccc(CC)s2)=O)=O)CC(NC(C2CN(C)C2)=O)CC(C)C1 Cc1nn(C)c(Cl)c1CC(=O)NC1CN(C(c2ccc(F)c(F)c2)=O)CCC1C N1(C(CCc2onc(C)n2)=O)CCN(C(c2ccoc2C)=O)CC(O)C1 CCC(O)C(C)C(=O)NCC1CC(O)(CNC(c2cccc(CCO)c2)=O)C1 C1(C)(C(=O)NC(C(=O)NCc2c(C)ccs2)CC2CCC2)CCOCC1 C1(C(=O)NCC=CCC(=O)N(CC(CC)O)C)CC2CC1CC2=O C1(CNC(CN(C(=O)CC(C)n2cccc2)C(C)C)=O)OC(=O)NC1(C)C N1(C(CN2C(C)CCC2)=O)CCN(C(c2cc3cscc3s2)=O)C2(CC2)C1 C(Cn1cccn1)(C(=O)NOCC1CCOCC1)NC(=O)Cc1ccon1 C12(CNC(c3ccc(C)s3)=O)CCC(C1)N(C(c1ccc(Br)o1)=O)C2 c1(NC(c2cc(Br)ncc2Br)=O)cccc(F)c1C(=O)Nc1nc(Cl)cnc1Br c1(C(N2CCCC(CN(C(C3(C)ON=C(C)C3)=O)C)C2)=O)c(C)nn(C)c1Cl C(=O)(C(C)C1=CCCC1)N(C(CNC(c1c(F)ncc(OC)c1)=O)C)C C12(C(NC(C(=O)NCC(C)(C)C(C)C)=O)C(C)C)CCC1CCN2 N1(C(c2c(C)coc2)=O)CC(NC(c2cnn3c2OCCC3)=O)CCC(O)C1 N1(C(C(C=C)CC)=O)CC2(CCCC2)C1C(=O)NC1CCC(F)(F)C1 C(=O)(CC(C)C(F)F)N(CC(C)NC(C1CCCN1C(=O)OC)=O)CC N1(C(c2ccc(CSC)o2)=O)CCC(CO)C(NC(=O)CN2CCOCC2)C1 N1(C(C(CSC)O)=O)CC(C(=O)NCCCN2CCOC2=O)CC1(C)C CON(C)CCN=c1nc2sccc2c(N2CCCC(c3n[nH]c(=N)o3)C2)[nH]1 N1(C(Cc2c(C)nc(C3CC3)s2)=O)CCN(C(=O)C(F)n2ccnc2)CC(O)C1 N1(C(C(C)(C)N(C)C)=O)CCC2(CC1)CC2CNC(c1cc(C(F)F)n(C)n1)=O N1(C(C(C)C(=O)OC(C)(C)C)=O)CCN(C(C2(O)CCOCC2)=O)CC1CF C1(NC(C(CCCNC(C)=O)(C)C)=O)CN(C(=O)Cc2ccco2)CC2(CCC2)C1 C1(C(N(CCSC)C)=O)CN(C(=O)C(C)(C)C)CC1(F)F c1(OC)ccc(CC(=O)NC(C2CN(C(C3CCCOC3C)=O)C2)C)c(C)c1 C12(NC(C=NOC)=O)CCC(CN(C(=O)C(C)Oc3cccc(C(C)=O)c3)C1)C2 c1(Cn2ncc(OC3CC(n4cc(-c5ccccc5)nn4)C3)c2)nnc(C)o1 c1(OC)cc(CNC(CS)C(C)C)cc(Br)c1O c1(C(CC)C(=O)NCCCN2CCCC2C(N)=O)ccc2c(c1)OCO2 CCC(CCCC(=O)N1CC2CCC2(C)C1)NC(c1cnnn1C)=O n1(CC(=O)N(C2(CC(N3CC4CC4C3)=O)CC2)C)cc(Cl)cn1 C1(C(C#C)NC(C2CCN2C(=O)CSCC(N)=O)=O)CCCCC1 CCCCC(CC)CC(=O)N(C1CCCN(C(c2cc(C(C)=O)c[nH]2)=O)C1)C c1(C(N2CC(CNC(CNC(C)=O)=O)CC2(C)C)=O)ccc2c(c1)OC(F)(F)O2 Cc1nc(C)c(CC(=O)N(C)CC2COCCN2C(=O)CC2CNC(=O)N2)s1 N1(C(C2ON=C(C(C)C)C2)=O)CCC2(CC1)CCN(C(C1CC(=O)N1)=O)C2 C1(C(=O)NCC(C2CCN(C(=O)CCCF)CC2)C)Cc2ccccc2C1 Brc1ccsc1CCCNCc1cnco1 N1(C(C2CC(O)(CNC(=O)CC(F)(F)C(F)F)C2)=O)CCCC2(CCOC2)C1 C1(C)(CC(=O)NCC(C)Cc2cn[nH]c2)CCN(C(=O)C=Cc2cc[nH]c2)C1 CCCCCCCCCC(O)C(=O)NCCCNC(=O)C1=C(Cl)CCC1 c1(C(N2CCC(O)(CCNC(C(C)=CC3CC3)=O)C2)=O)ccccc1P(C)(C)=O c1(C(=O)NCC(C(C)C)NC(C2CC(CC)OCC2)=O)ccn2c(C)cnc2c1 N1(C(Cc2c(C)cc(Cl)nc2)=O)CCCN(C(C2CC(C(F)F)C2)=O)CC1CO c1(C(C)C)cc(C(=O)NC2CC(F)(CNC(=O)CC(C)c3ccco3)C2)n(C)n1 N1(C(C(CN(CC)CC)F)=O)CCC2CC1CN(C(=O)C(C)N(C)C(C)=O)C2 C1(CNC(CCCCOC)=O)CCC(C)N(C(=O)COCCO)C1 c1(CC)nc(CCC(c2nnnn2-c2ccccc2)CCOC)no1 C(=O)(C1=CC2CCCCC12)NCC(CC)NC(c1ccc(F)cc1C(F)F)=O c1(CCC(N2C(CNC(=O)CC3(O)CCC3)CC2)=O)ccc2ccccc2n1 c1(NC(C(C)(C)CNC(=O)Cc2cccs2)=O)cccc2[nH]ccc12 c1(CNC(=O)NC(COC(=N)O)Cc2ccccc2)ccc(O)cc1Cl c1(C(N2CC(C(C)NC(Cc3c(C#C)cccc3)=O)C2)=O)c(C)ccc(F)c1N CC1=C(C(=O)NC(C)C(CO)NC(=O)Cn2cc(C(C)O)nn2)CCO1 N1(C(C2ON=C(CC)C2)=O)CC2(C=C(C(=O)N(C)CCC3CCCN3C)CO2)C1 c1(C(N2CCC(N(C(=O)COCCOC)CC)C2)=O)cnc2ccccc2n1 CC(Cc1cnn(C)c1)C(=O)NC(C)(CNC(=O)Cn1cnc(Br)c1)CO C1(NC(CC(=O)NCC2CC2)=O)CN(C(=O)CCC2CCCO2)CC1C1CC1 n1(CC)ncc(Cl)c1C(N1CC(NC(c2cscc2OC)=O)C(C)C1)=O c1(OCC)cc(CN2CC(O)CC2C(=O)NC(c2nccs2)C)cc(Br)c1O CC1CCCCC1(C)C(N1CCC(F)(C(=O)NCCc2ccccc2)C1)=O N1(c2cc(NCc3cncc(C=C)c3)ncn2)CCc2ccc(F)cc2C1 CON(C)C(=O)C(C)NC(N1CCCC(C2(C)COC(=O)N2)C1)=O c1(NCCN(CCCC)C)[nH]c(=NCCc2cc(F)cc(F)c2)nc2sccc12 c1(C(=O)NCCC=CC)nc2nccc(C)n2n1 Cc1nc(CC(=O)NCC2(NC(c3oncc3C)=O)CCC2)c(Cl)s1 NS(=O)(=O)c1ccc(NCc2ccc(O)cc2F)cn1 c1(SCC2CCC(C)(C)CO2)noc2ccc(Br)cc12 c1(C(=O)NC(C2N(C(C(CC)F)=O)CCC2)C)ccc(N2CCCCCC2)cc1 N1(C(COCCCCC)=O)CCCCC1C1CCN(C(=O)CC(C)COC)CC1 n1(CC2(C)CCCO2)c(-c2ccc([N+](=O)[O-])o2)csc1=NCCC(N)=O N1(C(C2(CC#C)CC2)=O)CCCCC(NC(=O)C(Cc2cnc[nH]2)NC(C)=O)C1 C(=O)(N=c1cc(C2CC2)n(C(C)(C)C)[nH]1)C1(C)CCN(C(C=C)=O)CC1 c1(C(=O)NC(C2CN(C(C3(C)CC(=O)C3)=O)C2)C)cnnc(Cl)c1 CC(CCC(C)(C)C)C(=O)NCC(C)(O)CNC(c1cc2nc(F)ccc2o1)=O C1(N(C(=O)C(F)(F)C2(O)CCC2)C)CCC(NC(=O)C(F)OC(F)(F)F)CC1 C12(CNC(C(C)N(C)C)=O)COCCN1C(=O)CN(C(c1cccnc1)=O)C2 C1(Nc2cc(OC)nc(C(C)C)n2)CC2CCC(C1)N2C(C1CCC2CC2C1)=O N1(C(C2(CC)COC2)=O)CC2(CC(NC(=O)C(c3ccccc3F)C)CO2)C1 N1(C(Cc2c(C)non2)=O)CCC(NC(=O)C(C)SC(C)C)C1C(C)C C(=O)(CC(C)(C)Cc1ccc(Cl)cc1)N1CCC(NC(CC2CN(C)C2)=O)C1 N1(C(c2cccc(C#C)c2F)=O)CCCC2(C1)CN(C(=O)CC1CCOC1C)C2 CC(Cn1ccnc1)C(=O)Nc1nnc(N2CCCCC2)s1 C1(=CC(=O)N(C(C(=O)N(CC(F)Cl)C)C2CC2)C)CCOCC1 C1(C(N2CCSC2c2ccc3c(c2)CCC3)=O)C2C3CC1C(F)(F)C23 c1(C(N)=O)cc(CC(=O)NCC2CCCCN2C(C2CC(O)C2)=O)cc(F)c1 c1(-c2c(OC)cnc(F)c2)c[nH]c2ncc(C(=O)Nc3cnn(CCO)c3)cc12 c1(OC)ccncc1C(=O)NC1CN(C(=O)Cc2ncccc2C)CC1C CC1CN(C(=O)CCC(=O)N2CCCC2)CC1NC(C1CC=CCC1C(N)=O)=O C#CC1CCCCC1OC(=O)CC1CCCC(C)(C)O1 C1(C(=O)NCCC2CCC2)CC2CC2N1C(=O)C(F)F N1(C(c2cc(CC(C)C)nn2C)=O)CC2(CCC2NC(=O)C(F)OC(F)(F)F)C1 c1(C(=O)NCC(CC)OC(C)C)nc(NC(=O)C(C)NC(N)=O)ncc1Br c1(CC(N2CC(NC(C(CC)C)=O)(COC)C2)=O)c(C)n[nH]c1C c1(C(N2C(CN)CCCC2)=O)nc(=NC2CC2)cc[nH]1 N1(C(C(F)=C(C)C)=O)CCC(NC(c2csc(C(F)(F)F)n2)=O)C(F)(F)CC1 C(=O)(CC(C)(C)O)N(C1CCN(C(C2(c3ccccc3)CCSC2)=O)C1)CCC c1(C(CC)C)nccc(=NCC2CN(C(c3cc(OC)cnn3)=O)CCC2C)[nH]1 c1(CNC(c2cncs2)=O)cccc(CNC(C2CCCCC2C(F)F)=O)c1 C1(C(N(C(C)CCNC(C2CC2(C)C(F)F)=O)C)=O)CC2(CC(=O)N2)C1 c1(C(=O)NCC(C2CCC2)NC(C(CC)(C)O)=O)ccc2c(c1)N(C)CC2 CCCCC(CC)C(=O)N(C1CCN(C(=O)CC2(C)CC2)CC1)CC1CCCO1 N1(C(C(C(CC)O)C)=O)CCC2CCC(C1)N2C(c1ccc(NC=O)cc1)=O C=C(Cl)C(C)(C)C(=O)N1CCN(C(=O)C(C)CCOC)C(c2cn[nH]c2)C1 N1(C(CN2C(C)CCCC2)=O)CCCC(F)(CNC(C2CC=CCC2)=O)CC1 [N-]=[N+]=Nc1ccc(C(=O)NCCNC(C2(C#N)CC3CC3C2)=O)cc1 O=C(CN1C(=O)Cc2cc(F)ccc21)NC12CCC1CN(C(c1cnco1)=O)C2 c1(C(=O)NCCC(C)N(C)C(c2cc(Cl)ccc2O)=O)ccnc2ccnn12 C1(C(N2CCC(NC(C(CC=C)CC)=O)C(CO)C2)=O)Cc2ccccc2C1 C=CC(C)(O)CC(=O)N1CC2(CNC(=O)C(SC)SC)CCC1C2 C(CCN(C(=O)C(O)CC1CCCC1)C)(C(C)C)NC(c1cc(C)on1)=O c1(C(N2CCC(NC(c3c(C)nc(CC)o3)=O)C(C)C2)=O)ccc(N)c(F)c1F CCC(C)C(O)CC(=O)NC1CC(N(C)C(c2n[nH]c(C3CC3)c2Cl)=O)C1 N1(C(c2c(C)nns2)=O)CCC(C)(C)C1CC(=O)N(CCS(C)(=O)=O)C C1(C(N2CC(CCNC(c3cnc(C)nc3C)=O)C2)=O)CCc2cnc(C)n2C1 N1(C(c2nc(C(=O)Nc3ccnc(C(=O)O)c3)sc2)=O)CCCCC(F)(F)C1 N1(C(CC(C)SC)=O)CCN(C(=O)C=Cc2cocn2)CC1CCO Cc1cc([N+](=O)[O-])c(C)cc1NCc1ccc(-c2ccc(SC(C)C)cc2)nn1 C(=O)(C(O)C1=CCCCC1)N1CCCC(N(C(C(=O)NCC(F)F)=O)CCO)C1 C(=O)(C(C)(C)C(C)NC(=O)OC(C)(C)C)N1CC(C)C(N2CCOCC2)C1 c1(N2CC3C(CNC(C(C4CCC(=O)N4)C)=O)C3C2)nc2cc(Br)cnc2s1 CCC(CC)CCCC(=O)NC1CCN(C(=O)CNC(=O)C(CC)CC)C1CC n1(-c2nc(C)cc(C)n2)[nH]c(=NC(=O)NC2CC3CC2C3)cc1C Cc1csc(C(=O)NC2CCN(C(=O)C(C)NC(c3ccccc3)=O)CC2)c1C CCC(C)(C)C(O)C(=O)NCC1CCCCN1C(=O)COCCCC(C)C CCCCC(C(=O)Nc1cc(CC)cnc1O)NC(=O)CC1CCC(O)C1 CC1CCCCC1(CNC(C1C=CC=CC=C1)=O)NC(c1cccnc1Cl)=O C#CCCCCCCC(=O)NCCC(=O)N(C)Cc1nccn1C(C)C C1(CC(=O)NC2CC(CCNC(C(C)(C)n3cccn3)=O)C2)CCCCC12CC2 C1(C(=O)OC)C=CCCN1C(C1COC(C)C1)C(=O)NCc1cccs1 C1(NC(C2(OCC)CCOC2)=O)CN(C(=O)CCNC(=O)OC)CC(C)(C)C1 Cc1cc2c[nH]nc2cc1C(N1CCC(F)(CNC(=O)CC2CCCCO2)C1)=O N1(C(c2c(C)ocn2)=O)CCCN(C(c2cn(C)cc(Br)c2=O)=O)CC1C c1(NC(C2CCN2Cc2cccc(-c3ccccc3)n2)=O)cc(O)nc(O)n1 c1(CNC(C(=O)NC(c2ccccc2F)C)=O)ccnc(C#N)c1 C1(C(=O)NC2C3CN(C(C(COC)(F)F)=O)CC32)CCCC2(CCC2)O1 Cn1nc(CNC(C2CC(CC(C)(C)C)C2)=O)c2c1CCN(C(=O)CO)C2 Cn1ncc(C(N2C3CCC2CN(C(=O)CCc2ccsc2)C3)=O)c1S(C)(=O)=O c1(C(N2CC(OC)C(NC(c3coc4c3CSC4)=O)C2)=O)cccn2nnnc12 c1(C(=O)NCC)cc(NC(C2CC(NC)CCO2)=O)c(C)s1 c1(C(=O)NCCN(C(=O)CC2CCCCC2)C(C)C)ccc(=O)n(CCO)c1 C=CC1(O)CCN(C(C2(SC)CN(C(=O)C(F)C(C)(C)O)C2)=O)C1 N1(C(C2N(C(CN3C(=N)NCC3)=O)CC(F)(F)C2)=O)CCC2CCCOC2C1 c1(NC(=O)NCc2c(OC)cncc2)nc2c(s1)CCCC2(C)C Cc1ccc(Sc2oc(C(N3CCCC(NC=O)CC3)=O)c(CN(C)C)n2)c(Br)c1 C(CCF)(C(=O)N1CCOC(CF)C1)NC(c1ccnnc1)=O C1(NC(c2cnn(CC(C)C)c2C(F)F)=O)C2Cc3c(Cl)cccc3C12 C1(NC(Cc2c(C)noc2)=O)CN(C(=O)CCN2CCCCCC2)CCC1CO c1(OC)cc(-c2nnc(C3COC4(COC4)C3)o2)ccc1CCO c1(C(=O)NCCC(C(=O)NC2C3COCC23)OC)cc(C)cc(C)n1 C1(NC(C2N(C(C(CSC)O)=O)C(C(C)C)CC2)=O)CCOCC12CCC2 C1(C(=O)Nc2nnc(OC)s2)(CNC(c2ccc(CSC)cc2)=O)CC(C)(C)C1 CC1CN(Cc2cc(C(C)(C)C)n[nH]2)CCC1NC(=O)CN(C1CCCCC1)C C(C(CC(=O)N=c1nc[nH]n1CCO)NC(=O)OC(C)(C)C)OC N1(CC2CN(C(=O)CC3C=CCCC3)C2)CCN(C(C23C=CC(CC2)C3)=O)CC1 C1(NC(c2c(C)ncn2C)=O)CN(C(c2ccc(F)cc2)=O)CC2(CCC2)C1 N1(C(COc2cccc(CC)c2)=O)CC2CC(F)(F)C2C1 CC(C)(CCCNC(=O)C=C1CCOCC1)C(=O)NOCC(=O)N(C)C C1(C(N2C(CNC(=O)CCCn3cccn3)COCC2)=O)CN2CCCN1CC2 C(=O)(C1=COCCO1)NCC(C)(C1CCC1)NC(c1c(C)csc1)=O C(=O)(CCCS(C)(=O)=O)NCC1C(NC(c2n[nH]c(C)c2Cl)=O)C1 C(C(O)CN=c1[nH]cncc1Br)NC(C(c1ccc(C)cc1)C)=O C(C(CC(C)C)NC(c1cc(=O)n(C)o1)=O)NC(c1ccc(CCC)s1)=O c1(C(C)C)nnnn1CC(=O)NC1CC(N(C(=O)CCCN2CCCC2)C)C1 Cc1cc(=O)c(C(N2CCN(C(c3ccc(Cl)c(N)c3)=O)C(C)C2C)=O)cn1C C(=O)(C1CCCc2sc(C)nc21)N1CC2CC(NC(COCCC)=O)C2C1 C(=O)(CCC(C)c1ccccc1)NCCN(C(c1c(NC)scn1)=O)C1CC1 C1(C(=O)NCC2(CO)CCN(C(=O)C3=CCOC3)C2)CC2OC1C1CC21 Cc1ccc(C)c(C(=O)NCC(CC(C)C)NC(=O)CC2CC23CC3)c1 C1(NC(CCC=C=C)=O)CC(O)CN(C(=O)COc2ccc(C)cc2F)C1 c1(CC(=O)N(C(C)CNC(=O)C(C)OCCOC)CC)n[nH]cc1C c1(CC(C)C)ccc(CC(=O)NCC(O)CNC(C2CNC(=O)N2)=O)cc1 C1(NC(=O)CCCc2ccsc2)CC2CC1N(C(C13COC(CF)(C1)C3)=O)C2 C1(C(=O)NCc2ccc([N+](=O)[O-])[nH]2)CCC2(CN(C(=O)C(F)(F)Cl)C2)O1 C1(NC(c2ccnc(C)n2)=O)CCN(C(=O)COCc2ccccc2C)CC1F c1(CC)cc(C(=O)NC2COCCN(C(=O)CC(C)(C)O)C2)cc(Cl)c1 C(C)(N=c1[nH]nc(-c2ccccc2)o1)C1CCN(C(c2cc(C)c(F)nc2)=O)C1 c1(C(=O)NC(C2CCCN2C(c2csnc2Br)=O)C)ncc(F)cc1N N1(C(CN2CCC(NC(CC3CN(C(CC)CC)C3)=O)C2)=O)CCCOCC1 C=CCCCCCCC(=O)N1CC(NC(=O)CCC(C)(C)F)C2CC12 C1(NC(C2CN(CCOC)C(=O)C2)=O)CC(C)CN(C(=O)Cc2cc[nH]n2)C1 C12(C(N3C(C(=O)OC)CCC3)=O)CC(CN(C(c3cc(C)sn3)=O)C1)C2 Cc1nc2cccc(C(=O)NCC3(C)CCCC3NC(=O)Cc3cc[nH]c3)c2[nH]1 CC(C)CC(C(=O)NC1CC2CCC(C1C)N2C(C1(C(C)C)COC1)=O)C(N)=O c1(OC)ccc(-n2nc(-c3occc3C)nc2CCC(C2CC2)C2CC2)cc1 C(=O)(C(C)(C)CC(=O)NCCCCC(C)NC(=O)C(F)C(F)(F)F)OCC Cc1cc(C(N2CC(CC(=O)NCC(C)(O)C3CC3)C3(CC3)C2)=O)cc(C#N)c1 N1(C(COCC(=O)NC)=O)CCC(NC(C2CCC(C(=O)OC)O2)=O)C(C)(C)C1 c1(C(=O)NC2CCN(C(c3cn(C)[nH]c3=N)=O)CC2O)cc(=O)n2ccsc2n1 CC1(C)C(=O)NCC1NC(C1CCC(CNC(c2c(I)ccnc2F)=O)CC1)=O N1(C(C2(N(C(=O)Cc3cccnc3O)C)CC2)=O)CC(C)(C)CCC1CO C(=O)(CCCC(=O)NC1(CNC(C2CC2Cl)=O)CCCC1)c1ccc(OC)cc1 N1(C(C2OCCN(C)C2=O)=O)CCC(C)(C)C(NC(c2cc(C(N)=O)cs2)=O)C1 Cc1nc(C(=O)NC2(CNC(=O)CCN3CCCC3)CC(F)(F)C2)sc1C C(=O)(C(C(C(C)C)C(C)C)N(c1ccc(F)c(Cl)c1F)C)NC(CC)C Cc1ccc2c(C(=O)NCC(C)N(C)C(c3cnc(C(N)=O)s3)=O)csc2c1 c1(C(c2n(CCCC)nnn2)NC(C2(n3ccnn3)CC2)C)c(Cl)cncc1Cl c1(C(N2CC(C)N(C(c3cc(F)cc(N)c3F)=O)CC2)=O)c(Cl)ccc(F)c1F CCC(C)(C)CCCC(=O)NC1CCCCC1NC(c1cncc(Cl)c1Cl)=O N1(C(c2c(Br)cn(CC)n2)C(=O)NCC2CC2)CCC2(CC(F)C2)C1 c1(C(=O)NCC2(F)CN(C(C=CC(=O)OCC)=O)C2)sc2ccc(C)cc2c1C C1(OC)CCCN(C(=O)C(C2CCC2)NC(=O)CCCNC(C)=O)C1 c1(C(=O)NCC2N(C(C(CCC)C)=O)CCCCC2)cccc2c1NC(=O)CO2 C#CC1(C(=O)N(CC(C)CO)C)CN(C(=O)C(F)CCC)C1 c1(C(N(CC(C)NC(=O)CNC(C)=O)CC)=O)cc(F)c(F)c(F)c1 c1(C(=O)OC)c[nH]ccc1=NC1CC(NC(=O)COCC2CCCO2)C1 c12ccnc(c1)Cc1cn-2nn1.C(C(C)C(=O)NC1CCCC1C(=O)O)SC CC(C(=O)NC1CC(NC(c2ccc(Br)c(O)c2)=O)C1)S(C)(=O)=O N1(C(=O)NC(C)Cc2c(Cl)cccc2Cl)CCC2(CCCNC2=O)CC1 c1(SC)ncc(C(=O)NCC2CC(NC(=O)C(C)C3=CCCC3)C(O)C2)c(O)n1 C1(CC)CN(C(=O)C(F)(F)c2ncccn2)CCN1C(c1ncc(N)cc1C)=O N1(CC2(CC)CC2)CC(C(=O)OC(C)(C)C)C(c2ccccc2)C1 C(=O)(C(C)S(=O)(=O)C(C)C)N(C1CN(C(c2ccc(F)c(C)c2N)=O)CC1O)C CCC(CC(F)F)C(=O)NC1(C)CC(NC(=O)CSc2ccc(Cl)cc2)C1 c1(OC)ccc(C(=O)NCCN(C)C(C2CC(SC)C2)=O)s1 c1(OC)ccc(S(=O)(=O)NCCc2ccc(-n3cnnn3)cc2)c(OC)c1C c1(C(=O)OC)ccc(NCC2CCN2C(=O)CC2CCCOCC2)c(C#N)n1 CC(C)C(C(=O)NC1CCCC1CN=[N+]=[N-])NC(=O)CC1CCOC1(C)C c1(CC)ncnc(N2CCSC(C(=O)NCC(C)(F)F)C2)c1F c1(CC)ccc(NC(=O)NC(CC)C(O)CC)c(Br)c1 O=C1CCCc2nc(NC3CS(=O)(=O)CC3NC(c3cncc(F)n3)=O)ncc21 c1(CC(=O)NC2(c3cn(CCS(N)(=O)=O)nn3)CCCCC2)cc(F)ccc1Cl C1(C(N(C(C)C)CCNC(c2cn(CCC(C)(C)C)nn2)=O)=O)COCCN1C c1(C(=O)NC2CCC(CNC(c3cc(N(C)C)ncc3)=O)C2)occ2c1CCC2 C1(CC)CN(C(=O)CC2CCC=CCC2)CCN1C(=O)C=C(Cl)Cl CCCC(CCC)C(=O)NC(CNC(C1C(C(C)=O)C1(C)C)=O)C1CC1 c1(NC(c2scc(C)c2C)=O)cc2c(cc1F)NC(=O)CC2 Cc1ccc(C(=O)NCCCC(C)(C)NC(c2cnc(O)cc2C)=O)c(N)c1 c1(C(N2CCC(CCC(=O)N(C(C(C)SC)C)C)CC2)=O)coc2ccccc12 CC1CN(C(c2cc(F)n(C)n2)=O)CCCN1C(=O)CC1CCCC(=O)N1 C12(NC(CC3CC(OC)C3(C)C)=O)CCCCCC1N(C(C1C=CCC1)=O)CC2 C1(CN(C)C(c2cc(-n3cc(N)cn3)ccn2)=O)CCCC2CC12 N1(C(CCSCC)=O)CCC(C)N(C(=O)CC(C)C(F)F)CC1 C1(C(=O)NCc2ncc(CC)[nH]2)CN(C)CCN1C(c1cc2n(n1)CCO2)=O C1(C(C)NC(c2n(CC#C)ccc2)=O)CCCCN1C(c1cscc1Cl)=O CCC(C(=O)NC1CCC(C(=O)NC2(CO)CCSC2)C1)SC N1(C(CCCOCC=C)=O)CCC(C)C(CC(=O)N(C)Cc2nccs2)C1 c1(C(=O)NCCCN(C(CCN(CCC)C)=O)CC)ccnc2ccc(F)nc12 N1(C(C(C)C2CCOC2)=O)CC(C2(NC(c3cnc(O)c(Cl)c3)=O)CC2)C1 CCC(C(=O)NCc1ccncc1)NC(=O)CC(C)n1cccn1 C1(c2n(CCC)nnn2)(NC(C)CNC(=O)OC(C)(C)C)CCC(CC)CC1 C(=O)(C(F)(F)Cc1ccccc1)NCC1(c2cn(C)nc2)CC1 C1(CC)CN(C(=O)COCC2CCC2)CC1C(=O)NCC1(C2CC2)CC1 CC1CCN(C(=O)Cn2cnnc2O)CC1NC(C1(CS(N)(=O)=O)COC1)=O C12CCCC1C(=O)NC2.C1(CC)CC(CC(=O)N(CCCN2CCCC2)C)C1 c1(C(=O)NC(CNC(Cc2c(C)n(C)cn2)=O)C2CC2)cncc(O)c1Cl O(N1C(=O)c2ccccc2C1=O)C(CCOC(C1CC2CCC1(F)CC2)=O)=O CC(C(=O)NCCOC1CCN(C(c2csc(C(F)(F)F)n2)=O)C1)P(C)(C)=O C#Cc1ccc(C(N2CC(C(=O)N(C3CC(OC)C3)C)C3(CC3)C2)=O)cc1C CC1CC(C#N)(C(=O)NC2CCC(NC(c3ccc(CO)o3)=O)CC2)C1 C1(CC)(CC)CCN(C(C23CC2CCN3C(c2ccc(C)o2)=O)=O)CC1 c1(CC)ccc(NC(C2CN(C(c3[nH]cnc3C)=O)CCO2)=O)cn1 C(N=c1[nH]c(=NC2CN(C3CCC3)C2)[nH]c2c1COC2)c1c(C)cc(C)cc1C c1(C(N2CCC(NC(c3c(C)n[nH]c3C)=O)C2C)=O)cn(C)ccc1=O C1(NS(NC)(=O)=O)CCN(C(C2(Cl)CCCCC2)=O)CC1 c1(CC)cc(C(=O)NCC2CCCC2NC(=O)Cn2nnnc2C2CC2)nn1C c1(C(=O)NC2C(NC(C(C)=C3CCC3)=O)CC2)cc(-c2cccnc2)on1 CN1CCN(C(C2CC(=O)OC2(C)C)=O)C(C(N2CCOC3CCC23)=O)C1 C1(NC(CN(C)CCOc2ccccn2)=O)CC(N=c2[nH]ccn3ccnc23)C1 C(CC(=O)N1CCN(C)CC1C)(C(C)C)NC(c1cc(CC)on1)=O N1(C(CC)=O)CC(C)CN(C(C2CCC(C)(O)CC2)=O)CC1C c1(C(=O)NCCN(C(=O)CC2CCC(C)CO2)CC)c(F)ccc2ccoc12 c1(OC)cc(C(C)(C)NC(=O)CNCc2ccc(O)cc2)cc(F)c1O c1(N2CCC(N(C(C)=O)C3CC3)C2)ccc(S(=O)(=O)N2CCCC2CO)cn1 C(CCCN=c1[nH]c(=NC2CCC3CC23)c2c(ncn2C)[nH]1)n1c(C)ncc1 c1(CNCC2OCCC(NC(=O)OC(C)(C)C)C2)ccn2ccnc2n1 C1(NC(c2n(C)nc(O)c2)=O)C2CC(CN(C(=O)Cn3nnc(=O)[nH]3)C2)C1CO N1(C(c2c(CC#N)ccs2)=O)CCCC(NC(=O)C(F)(F)c2cncs2)CC1 N1(C(CC(CC)C(F)F)=O)CC2(CCCN(C(C3CSC3)=O)C2)C1 Cc1cccc2c(C(N3CCN(C(c4ccncc4O)=O)C4CC34)=O)cnn12 c1(C(=O)NC2CCN(C(c3cccc(CC)c3O)=O)CC2)cc(C)c(C)cc1N c1(C(N(CCNC(c2c(C)nnn2CC)=O)CC)=O)cn(C)c(=O)nc1O c1(C(=O)NCC(N(C(C=C(CC)C)=O)C)C2CC2)cc2cccc(C)c2s1 c1(C(N(C2C(O)CCN(C(C(C=C)O)=O)C2)C)=O)ccn2nnnc2c1 C1(C(=O)NCC(C)(C)OCC(=O)N(C(CCSC)C)C)CCCCC1O c1(CNC(C(C)(C)C2CCCN2C(=O)CNC(N)=O)=O)ccncc1F CC#CC1CN(C(c2cnn(-c3ccc(Br)cc3)n2)=O)C1 CC1(C)CC(CNC(=O)Cc2cc(F)ccc2F)CN1C(C1CCS(=O)CC1)=O c1(C(N2C(CCNC(C3COC(=O)N3)=O)CC(OC)C2)=O)cc2n(n1)CCO2 c1(OC)cc(C)c(CC(=O)NCC(C)NC(=O)CC2CC(C)C2)c(C)c1 Cc1cc(Br)c(C(N2CCC(CCCN(C)C)CC2)=O)s1.N12CCCC1C2=O CC1C(NC(C2CCNC2=O)=O)C(C)CCN1C(c1cccn2nnnc12)=O N1(C(=O)CNc2c(C(C)=O)cccc2)CC(F)(F)CC1C(N)=O CCC(CC(=O)NCCCCN(C(=O)C(C)NC(=O)OC(C)(C)C)C)C(C)(C)C N1(C(C(C)c2cc[nH]n2)=O)CCC2(CC2)CC1C(=O)NC1CC2(CCC2)C1 c1(C(=O)NCC(CN(C(C2CC(F)C2)=O)CC)(C)C)cc(C#N)ccc1N C1(C(N2CCC(CC=C)C2)=O)(NC(c2cscc2CC)=O)CCN(C)C1 c1(CC)ccc(C(=O)NC2CCN(C(=O)C(F)CC3CC3)CC2O)c(Cl)c1 c1(C(N2CC(CNC(CC(CCC)(C)O)=O)OCC2)=O)ccn2cnc(C)c2c1 C1(CCCNC(C2(CCCC)CCC2)=O)CCN(C(C2(C)CCOC2C)=O)CC1 C(=O)(C1=CC(C)CC1)NC1CN(C2CN(C(CCC=C)=O)C2)C(=O)C1 N1(Cc2ccc(SC)c(Br)c2)C2CCCC1CC1(C2)NC(=O)NC1=O C1(C(N(CCC)C(C)C)=O)CCCC12CCN(C(=O)C(F)Cl)C2 Cc1nc(NC(=O)C(N)CC2CCC2)oc1-c1ccc(Cl)cc1 C1(N(C(CN(C2CC2)CC)=O)C)CCC(NC(=O)CC23CCC(CC2)C3)CC1 c1(C(=O)NC2C3CN(C(C(F)OC)=O)CC2C3)ccc2nc(C)[nH]c2c1 c1(SCCS(Cc2cn(CCCC(=O)OC)nn2)(=O)=O)oc2ccccc2c1C c1(CC(=O)NCC2(CNC(C=CC(CC)C)=O)CC2(F)F)nnc(S)n1C C(=O)(CC1CCc2ccccc21)N1CC(CNC(=O)CCCC2CCCC2)C1 C1(C(=O)NC2C(C)CN(C(=O)CC3OCCC3C)C2)CCC2CC2CC1 CC(C)CC(C)C(=O)NCC1CN(C(c2c(F)cncc2Cl)=O)CCN1C c1(CCC(=O)NC(CC(C)NC(COC)=O)C)cccc(N(C)C)c1 CC(C)C(C)(C)C(=O)NC1CC2CC(NC(=O)C(N3CCC(O)CC3)C)C1C2 CC(CS(C)(=O)=O)C(=O)N1CCCC(CO)(NC(c2cc(=N)[nH]c(Cl)n2)=O)C1 c1(NC(C2C(O)CCN2c2ccn3nccc3n2)=O)c(Br)ccc(F)c1F C(C)(C(=O)NC1CC(CC(=O)NCC2(C(C)(C)O)CCC2)C1)SC(C)C c1(Cn2cc(CN3CC(CC)OC(C)C3)nn2)nsc2ccccc12 N1(Cc2c(OC)nc(C)cc2)CCCC12CN(S(=O)(=O)Cc1ccc(Br)cc1)C2 C12(CNC(C3CNC(=O)N3)=O)CCC(C1)N(C(=O)COC1CC(F)(F)C1)C2 Cc1coc(C=CC(=O)N(C2CCCN(C(=O)C(C)n3cccc3)C2)CCF)n1 C(C)(CCC(=O)NC1(C(=O)NCC2CCCOC2)CCCC1)SC c1(OC)c(C)nc(C2CC2)[nH]c1=NCCC1CCN(C(c2nccn2C)=O)C1 C#Cc1ccccc1CC(N1CCC(C(=O)NCCC2CCCC3CC23)CC1)=O C(=O)(CC(C)C(F)F)N1C(CNC(c2cnc(NC(=O)C(C)C)s2)=O)CC(OC)C1 C1(OC)CN(C(c2ccc(C(C)C)c(Cl)c2)=O)C(C)(CNC(c2cccs2)=O)C1 N1(C(c2cc(OC)n[nH]2)=O)C2CCC1CC(C(=O)NCC1CC3(CCC3)C1)C2 Cc1sc2nc1C(=O)N1CCN(CC1)C(=O)c1cccc-2c1.C(C(C)(C)O)CCO C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CCC(C)(NC(Cn2c(C)ncc2)=O)CC1 c1(CNC(=O)Nc2nc(C)nn2C)cc(F)cnc1Cl N1(C(c2c[nH]c(=NC)s2)=O)CC(NC(c2c(C)ccnc2C)=O)CC(C)C1 C1(CC(=O)NC)CCN(C(=O)C(C)CNC(C2CC(CF)C2)=O)C1 N1(C(CCSC)=O)CCCC(c2n[nH]c(CNC(=O)C(C)NC(C)=O)n2)C1 C#Cc1ccc(OCC(=O)NCC2CCC(NC(C3CCNC3=O)=O)CC2)cc1 N1(C(c2c(C)n(C)nn2)=O)CCC2(CCN(C(C3CCCCC3N=[N+]=[N-])=O)C2)C1 C(CC(=O)NC(C)(CO)C(F)F)(C(F)F)NC(c1c(C)ncs1)=O N#CC1(C(=O)NCC2CCCC2NC(=O)CCc2ccccn2)CCSCC1 C1(NC(CN(C2CCC2)C)=O)CC(CNC(C2CC2(F)F)=O)C1 C#CCCC(O)C(=O)NCC1(COC)CN(C(C2CC2c2ccccc2F)=O)C1 N1(C(C(C)c2ccsn2)=O)CCCC12CCN(C(=O)CS(=O)(=O)CCO)C2 C1(NC(=O)CC2CC2C(F)(F)F)CCN(C(c2cscn2)=O)C12CCC2 C1(CC)C(=O)NCCCN1C(=O)CNC(=O)CNC(=O)C(C)c1cccs1 c1(NC(C2C(C(N(CC(F)(F)F)CC)=O)C2)=O)cc(C(C)(C)C)nn1C C(=O)(C(C)(C)CCCNC(=O)CCCF)N1CCCC(COC)C1 O=C1OC2C(NCC(O)COc3ccc(F)cc3)C3CC1C2C3 C(=O)(C1CCc2nccn21)NC1(COC)CCN(C(=O)CC2(O)CCC2)C1 N1(C(c2c(C)noc2C)=O)CC2(CC(NC(=O)CN3CCCCCC3=O)CO2)C1 c1(C(=O)NCCCCC(C)NC(=O)C2=CCSC2)cn(C)ccc1=O C1(NC(C2(CNC(C(CC)C)=O)CCCC2)=O)CC2CC(O)C1C2 c1(N2CCC(OC(F)F)CC2)[nH]c(=NCC2CC3CCC2CC3)nc2sccc12 c1(C(=O)NCC(=C2CN(C(CSCC=C)=O)C2)F)nc2ccccc2cc1C C(=O)(C(C)S(=O)(=O)C(C)C)NC1C2CN(C(c3c(C)ncn3O)=O)C1C(O)C2 N1(C(C(C)N(C(C)=O)C)=O)CCC(C)(C(=O)NOCCO)C1 c1(C(=O)NCC2N(C(C(F)(F)C3(OC)CCC3)=O)CC2)cnc2c(F)cccn12 Cc1ocnc1-c1cn(CCCCCNC(=O)Cc2csc(Cl)n2)nn1 c1(OC)nc(C(=O)NC2CC(NC(=O)C(C)COc3ccccc3)C2)co1 C1(C(=O)NCCCOC)CCCN1C(=O)CSC(C)(C)C c1(C(=O)NC(CC)CN(C(=O)C(O)Cc2cnn(C)c2)C)cccc2ccoc12 c1(C(CC)(C)C)ccc(C(=O)NCC2CCN2C(=O)Cc2ccc(C)nn2)cc1 N1(C(CC(=O)NCC#C)=O)CC2(CCN(C(C3C=CCCC3)=O)CC2)CC1C C1(NC(Cc2cc(C)[nH]n2)=O)CCC(O)CN(C(C2CC3(C2)CC(F)(F)C3)=O)C1 c1(C(C)OC(C)C)ccc(NC(=O)C(=O)NCC2CC3CC3C2)cc1 C(CCCCC(=O)NCCOCCCNC(=O)C(C)n1cccn1)OC Cc1c(C(=O)N(C(CNC(=O)CC2CCC(C)CC2)C2CC2)C)sc2nccn12 c1(C(N2CCCC(NC(C(C(C)C)OC)=O)CC2)=O)cc2c(nc1O)CCSC2 CS(=O)c1ccc(C(N2CC3(NC(c4cnn5c4NCCC5)=O)CC2C3)=O)cc1 C1(CNC(C(C)c2ccsc2)=O)CC2(CCN(C(=O)CCC3CC3(C)C)CC2)C1 c1(OC)ncc(Br)c(N2CCCC2CCCNC(c2ccc(C)n2C)=O)n1 c1(C(=O)Nc2cccc(C(N3C(C)CCCC3C)=O)c2)c(F)cc(F)cc1Cl C(CC(C)C)(C(=O)N1CCC(N(C(=O)C=C(C)c2ccsc2)C)C1)NC(C)=O N1(C(c2cc(OCC)ns2)=O)CC(OC)CC(NC(C2CC2[N+](=O)[O-])=O)C1 C(CCC(C)C)(C(=O)N(C1CCCC(O)C1)C)NC(c1cc(COC)on1)=O C(=O)(C(C(=O)NCCc1ocnc1CNC(c1cncn1C)=O)C(C)C)OCC CC1CC(CNC(c2cccs2)=O)CN1C(=O)C(C)CC1CCCO1 C1(CC)CN(C(c2coc(C3CC3)n2)=O)CCN1C(=O)C#CC(=O)N(C)C C(=O)(C1=CNC2=NCCC2=C1)NC1CN(C(C(CC#C)(C)CC)=O)CC1C C(=O)(CN=c1ccc(Cl)n[nH]1)N1CCC(CNC(c2ncc(C)cc2F)=O)CC1 CC1=C(C(=O)NC2CC(F)CN(C(=O)C(F)(F)C(F)F)C2)CCCO1 C=CCC(C(=O)N1CCC(CCNC(C23CCN(CC2)C3)=O)C1)C(C)C Cc1ccccc1CC(N1CC2CC2(NC(N2CCN(CC(C)C)CC2)=O)C1)=O N1(C(C2(CC=C)CC2)=O)CCC(C(C)CNC(c2cc(CC)sn2)=O)CC1 c1(NC(N2C(CCC=C)CCC2)=O)c(C#N)n(O)c2ccccc2[n+]1=O c1(N2CCN(Cc3c(F)cc(OC)c(F)c3)C3C2C3)ncc2c(ccn2C)n1 C(=O)(CCC(CF)CF)N(CC(CN(C(=O)CCC1CCCC(O)C1)C)O)C C1(CNC(C(CC)O)=O)CN(C(C23CC(C#N)(C2)C3)=O)CC1C C1(C(=O)NC2CC(CN3CCOCC3)C2)CC(=O)N(CCl)C1.c1(CC)ccccc1 Cc1ccc2c(C(=O)N(CC(C)NC(C3CCC(C)O3)=O)C)ccnc2c1C c1(CC)ccc(C=CC(=O)NC2CC(O)CN(C(c3ccco3)=O)C2)cc1 Cc1cc(O)cc(O)c1CN1CCCC(C)(C(=O)Nc2cccc(Cl)n2)C1 N1(C(CS(CC)=O)=O)CCC(CO)(CNC(=O)CCc2cnn(C)c2C)CC1 N1(C(c2cn(CC)nn2)=O)CC2CCN(C(c3cc(C)cnc3N)=O)CCC2C1 C1(O)(CNC(c2c(OC)csc2)=O)CCCN(C(=O)C=Cc2ccncc2)C1 c1(NCC(C)CC2(C)OCCO2)ncc(S(=O)(=O)NCC2CCCCC2)cc1Cl C(C(CC(F)(F)F)NC(C1(C)CC1(F)F)=O)NC(c1cn(CCOC)nn1)=O N1(C(c2n(CC)cc(Cl)c2)=O)CC2CCC2(CNC(C2CC(F)CN2C)=O)C1 O=C1CC2(CC(C(=O)NC3(CNC(C4CN(CC(F)(F)F)C4)=O)CCCC3)C2)N1 N1(C(C(C)OCC#C)=O)CCC(NC(c2ccc(C#N)o2)=O)C1(C)C c1(OC)ccc(CN2CCC2C(=O)Nc2nc(Br)ccc2Cl)c(OC(C)C)c1 c1(C(=O)NC2C3CN(C(C(C)O)=O)CC2COC3)c(Cl)cc([N+](=O)[O-])cc1Cl N1(C(C2ON=C(CC)C2)=O)CCC(NC(=O)CC2(CC(=O)OC)CC2)C(C)(C)C1 N1(C(C(CCC)C)=O)CCN(C(c2cc(COCC)cs2)=O)C(CS(C)(=O)=O)C1 C(=O)(C(F)(F)C(O)C(C)C)N1CC2CN(C(c3c(C)ccc(SC)c3)=O)CC2C1 c1(C(N2CC3C(NC(C(C(C)C)O)=O)C(CC3)C2)=O)ccc(S(C)(=O)=O)cc1 C1(NC(CC=C(C)C)=O)CC2CC1CN(C(=O)C(O)Cn1cncn1)C2 c1(CC)noc(CCCC(=O)N(CC(O)CNC(=O)CCc2cn[nH]c2)C)n1 C1(N(CC(c2ccc(O)cc2)O)C(C2CC2F)=O)CCC12CCNCC2 C1(CNC(c2sc(F)cc2Cl)=O)CCN(C(=O)CCOC2CC2)CC1(F)F C1(C)(CCNC(c2c(CC)n[nH]c2)=O)CCN(C(c2c[nH]c(=N)s2)=O)C1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCC1(NC(=O)C=Cc2cn[nH]c2)CCCC1 C1(C)(CC)C=C(C(=O)NCCC2CCCN(C(=O)Cn3nccc3C)CC2)C1 C1(C(N2CC3(CC(CNC(=O)CN4CCNC4=O)C3)C2)=O)Cc2ccccc2C1 C#CC1C(C(=O)NCC=CCNC(=O)C(C)OCc2ccncc2)C1(C)C c1(C(N2C(CCCNC(C3CC(C)(CC)C3)=O)CCC2)=O)cccc(C(N)=O)n1 N1(C(CCCSC)=O)CCC(CNC(C2CCC3CC3CC2)=O)CC1C Cn1c(C(=O)COC(C2CCCCC2c2ccc(F)cc2)=O)cnc1O N1(C(CSCC=C)=O)CCC2C(C1)CN2C(=O)C(C(C)C)n1cnnn1 N1(C(c2c(C)ccnc2)=O)CCC(CNC(=O)C(C)P(C)(C)=O)C(F)(F)C1 C1(CNC(C2CC2C(F)(F)F)=O)CC(O)CN1C(=O)Cc1cccnc1F N1(C(c2cn(CCCC)nn2)=O)CC2=C(C1)CN(C(C1(O)CC(CF)C1)=O)C2 C(=O)(C(F)C(F)(F)C(F)(F)F)N1CCCN(C(CC(C)(C)SC)=O)CC1C C1(N(C)Cc2cc(CSC)no2)CCCC(N)C1 c1(CC)nc(C)[nH]c1C(=O)NCCN(C(=O)C=Cc1scnc1C)C1CC1 N1(C(c2ccc[n+]([O-])c2)=O)CCN(C(c2csnc2Br)=O)C(CO)C1 N1(C(C(CC=C)NC(c2scnc2C)=O)=O)CCC(=C(F)F)CC1 N1(C(C(SC)SC)=O)CCC2(CC2C(=O)N(C)Cc2cncs2)C1 C1(COC)(CNC(=O)CCC(C)OC)CCN(C(=O)CCc2cccc(F)c2)C1 C1(C(=O)NC(CCC)C)C2CCCC2CN1C(c1oc(C)nc1C)=O c1(-c2cc(C)cc(C)c2)ccc(C(=O)NCc2cccc(CO)c2)c2[nH]ccc12 Cc1cc(C(N2CCCC2C#N)C(=O)NC2CCC2)c2c(c1)CCC2 N1(C(C(COCC)C)=O)CCCC(C(=O)NCc2snnc2C)C1 Cc1ccc(C(=O)NCCCOCCNC(c2ccc(F)cn2)=O)c(C)c1Br c1(CNC(C(CC(=O)OC)NC(=O)OC(C)(C)C)=O)nc(Cl)nc2c1COC2 c1(SC)c(C(=O)NCCCOCCNC(c2n[nH]cc2C2CCC2)=O)cnn1C N1(C(C23CCC2C3)=O)CCC(C(c2ccncc2)O)CC1 C1(C(=O)NCC2(C)CC(C)C2)CCCN(C(c2cc(O)nc(O)n2)=O)CC1 C1(c2n(CCSC)nnn2)(NCC2CCCCC2(C)C)CCS(=O)CC1 c1(C(N(C2CCN(C(c3ncc[nH]c3=O)=O)C2)CCC)=O)cnc2[nH]cncc1-2 C1(C)(C(N(CCN(C(C)C)C(C2CCC2(C)C)=O)C)=O)CCOC(C)C1 C12(NC(c3ccc(CO)c(F)c3)=O)CCCC1CN(C(=O)CCc1nncs1)C2 C12CC(=NO1)C(=O)NC2.Cc1cnn(CCC(=O)NCCSC(C)(C)C)c1 C#Cc1ccc(C(N2CC3(CC(NC(=O)C(C)OCCC=C)CO3)C2)=O)c(C)c1 c1(NC(C2(C)CCN(Cc3c(C)nc(C)[nH]3)C2)=O)ccc(OC(F)F)c(O)c1 CCCCCC(C)CC(=O)NC1(C)CCN(C(=O)CNC(=O)CCC(C)C)C1 c1(C(N2CC(C)N(C(C3CCSC3)=O)CC2)=O)ccnc2ccncc12 C1(C)(NC(c2ccc(OC)nc2C)C)CCC(C)=C(C)C1 C1(NC(=O)Cc2c(Cl)cccc2Cl)CN(C(C2CCOC2)=O)CCC12CCC2 N1(C(C2CC(NC(C3C(CC)OCC3)=O)C2)=O)CCC(C2CCC2)CC1 N1(C(=O)NC2CC(C)(NC(=O)OC(C)(C)C)C2)CCCSCC1C1CCC1 C(CCF)(C(=O)NC(C)CCC1CCCC1)NC(c1c(C)occ1)=O Cc1ccc(C(=O)NC2(CCCC(=O)N(C3CC3)CC3CCOC3)CCC2)o1 N1(C(C(C=CC)O)=O)CCN(C(=O)CCOC(C)CC(C)C)CC(C)(F)C1 c1(C(=O)NCCCCCn2cc(-c3ccsc3)nn2)ncc2cc(Cl)ccn12 c1(C(N2CCC(C(C)NC(c3cccc(Cl)c3O)=O)C2)=O)c(F)cc(F)cc1Cl C(c1ccccc1F)=CC(N1CCN(CCC2CC(O)C2)C2CC12)=O CN1C(=O)CCCC1C(=O)NCC1CCC1C(=O)NCCOCC(C)(C)O N1(C(c2cnc(OCC)nc2)=O)CC(NC(c2ccc(O)nc2)=O)C2CC2C1 c1(C(=O)NCCC2(NC(CCC3C(C)C3)=O)CCCC2)ncc([N+](=O)[O-])n1C C1(O)(CC(N2CC(NC(C(C)OCC)=O)C(OC)C2)=O)CCCCCC1 Cc1c(C(N2CC(O)CC2CNC(c2nnn(C)c2C)=O)=O)nc2sccn12 C(=O)(C(C(C)(C)C)C1CCC1)NCCC(C)NC(C1CC(C#N)C1)=O C=CCCCC(C(=O)NCc1nc(=O)o[nH]1)NC(C1CCC2(CCC2)O1)=O c1(-c2nnc(CCCC(N3CCC(SC)CC3)=O)s2)c(C)cccc1Br c1(C(COC(c2nc(CSC)sc2)=O)=O)cc2ccsc2n1C N1(C(C(C)OCc2ccc(F)cc2)=O)CCn2nnc(CO)c2C1 C1(C(N(CCNC(c2coc(-c3cccnc3)n2)=O)CC)=O)CCOCC12CCC2 c12c(cccc1Cl)OC(=O)C(C)C2=O.C1(NC(C)=O)CC(C)(NCC(=O)OC)C1 c1(C(=O)NCC2(OC)CN(C(=O)Cc3ncncc3Cl)C2)sccc1C#N CC1(C)C(CNC(=O)COC(C)(C)CNC(C2CC2[N+](=O)[O-])=O)C1(F)F C1(C(C(=O)NCCN(C(CC)=O)C2CC2)C)CCCCN1C N1(C(=O)OCC)CC2CCC1C(C(=O)NCC(c1ncccc1O)=O)C2 C1(NC(C(=O)O)C2CCCC2)CCC(N2CCN(CCC)CC2)CC1 Cc1cccc(Br)c1C(C(=O)Nc1ccc(O)c(Cl)c1)NC(=O)C=CC(=O)N(C)C CC(CCCNC(c1cscn1)=O)NC(c1ccc(CN2CCCCC2)o1)=O c1(C(=O)NC(C2CCN(C(C3(C)CCC(=O)C3)=O)C2)C)cc(O)ncn1 N1(NC(c2cnc(CN)s2)CC)CC(Oc2ccccc2)CC(C)C1 CC1CCCCC1(CNC(c1cc(Cl)on1)=O)NC(C1CSCC(=O)N1)=O N1(NC(=O)NC2N(C(c3ccc(Cl)nc3Cl)C)CC=C2)Cc2ccccc2C1 c1(C(=O)NCC2(C)CN(C(c3cc(F)c(Cl)nc3Cl)=O)C2)cc(Cl)c(F)c(Cl)c1 CCCCC(C(=O)N1CCCC(CCO)CC1)NC(c1occc1C)=O C(C)(C)(C(C)CC(=O)NCC1(C2CC2)CCCO1)NC(C1C=C(C)CS1)=O C1(N(C)C(C2CCCC2F)=O)CCCC(NC(C2C(C)(C)C2(C)C)=O)C1 c1(C(=O)NC(C)C(CO)NC(c2ccccc2)=O)cc2cc(Br)ccc2[nH]1 C(C(CNC(C1COCCO1)=O)C(F)(F)F)NC(=O)Cc1cc[nH]n1 C#Cc1cccc(CNC(c2ccccc2)C(F)F)c1 N1(C(C(C)CC#N)=O)C2CCC1CN(C(C13CC(F)(C1)C3)=O)C2 C(=O)(C(=O)C(CC)OC(=O)CCc1ccc(CC(C)C)cc1)OCC C(=O)(C(C)(C)C(=O)NC(CNC(c1c(C)cnn1C(C)C)=O)CC(C)C)OCC C1(NC(C(F)=C(C=CC)CC)=O)C2CC3CN(C(=O)CC4(CO)CC4)C1C3C2 c1(C(C)C)ncc(C(=O)NC2CCCC2NC(=O)CN(C2CCC2)C)[nH]1 C1(C(=O)NCCCC(C)c2ccccc2)CN(CC2CC3CC(=O)C2C3)CC(C)(C)C1 N1(C(c2ccc(OC)c(C(C)C)c2)=O)CCCC2CN(C(=O)CCF)CCC12 c1(C(=O)NCC(C2CCCC2)NC(C(C)(C)OC)=O)ccc2nccn2c1 C1(NC(c2cc(CN(C)C)on2)=O)CCCN(C(=O)C(F)n2cccn2)C1 C1(C(N(CCC(C)NC(c2coc(C(F)F)n2)=O)C)=O)CNC(=O)N1C CS(=O)(=NC(=O)C1CCC1)c1cnn2c1CN(C(C1CCC3(CCC3)O1)=O)CC2 C#CCCC(C(=O)NCc1nc(CCC)no1)NC(c1cn(C2CC2)nn1)=O C(C)(CC(N)=O)N(C(CC1CC(NC(CCC2CC(C)C2)=O)C1)=O)C CC1CCOCC1C(=O)NC1CC(CNC(=O)CNc2cccnc2)C1 N1(C(c2cnc(SC)[nH]2)=O)CCC(NC(c2cnn(CCF)c2)=O)CC1C c1(C(N(CCCC(=O)NC2C(C)(COC)CCC2)C)=O)cc(C)c(O)nn1 CN1CCCC(C(N2CCCCC2CN(C)C(c2cnccc2Cl)=O)=O)C1 C1(CNC(C(C)N(C(=O)C(C)CO)CC)=O)CC2CCCC2C1 c1(C2(C(N3CC4CC3CN4CC3CC3)=O)CC2)c(Cl)cccc1Cl CCC(C)C(C(=O)N1CCC(CNC(=O)C=CC2CCCC2)C(O)C1)NC(N)=O c1(C(=O)NCCCCC(C)NC(c2c(C)nc[nH]2)=O)ccc(F)cc1Cl N1(C(C(C(C)C)NC(C)=O)=O)CCC(C(=O)NCCCC(F)(F)F)C(O)C1 c1(C(C)=O)ccc(S(=O)(=O)N2CC3C(C2)N3C(=O)CCn2nc(C)cc2C)cc1 N1(CC)CCOCC1CC(=O)NC(CNC(=O)CC1CCCC1O)C(C)(C)C C(CCC(=O)N(CC(=O)NCCC1(C)CCCO1)Cc1ccccc1)NC(C)C C(CC(C)(C)NC(=O)Cc1cnc[nH]1)NC(C1C(C(N(CC#C)C)=O)C1)=O c1(OC)ccc(CC(=O)NC(C2CCN(C(C34CC5CC3C4C5)=O)C2)C)c(C)c1 C1(C(C)(C)C)CCN(C(=O)C(N2CCC(N3CCOCC3)C2)=O)CCO1 C(CCC(C)C)(C(=O)N1OC2C=CC1CC2)NC(C(CC=CC)CC)=O N1(C(Cc2c(C)ncs2)=O)CC(C)CN(C(c2nc(C3CC3)cs2)=O)C(C)C1 C1(C(c2n(CC3C(C)C3)nnn2)NC(c2cc(Br)cn2C)=O)C2CCOCC12 c1(C(=O)NCCC2CCC(NC(C(C)=CC3CC3)=O)C2)cc(C)nc2ncnn12 Nc1c(Cl)ccc(C(N2CC3(C2)CN(C(C2CC4CCCC(C2)C4)=O)C3)=O)c1Cl C(=O)(C(F)C(F)(F)F)NCC(C(C)C)NC(C(C)=C(C)C)=O C1(CNC(c2c(C)[nH]cc2)=O)CC(F)CN1C(=O)CCc1nccs1 N1(C(C(CNC(C2=C(C)CC2)=O)N(C)C)=O)CC2(CCN2C)C1 C(=O)(CCS(C)(=O)=O)NCCCN(CC(C)O)C(C)C C1(N(C(c2ccccc2)=O)CC)COCCN1C(c1cnc(-c2ccoc2)s1)=O c1(C(=O)NC23CC(CNC(CSCC=C)=O)(C2)C3)ccc(N)c(C)c1C c1(C(N(CC(C)NC(c2cc(C(C)=O)on2)=O)C)=O)cc(C)n(CC(F)(F)F)n1 c1(C(=O)NCC2CCN(C(C(c3cn(C)nc3)O)=O)C2)cc2c[nH]nc2s1 CCCCC(C(=O)NC(CC)C(=O)NCCC)NC(=O)CC1(O)CCCCC1 c1(NC(=O)NCC(C2CCCOC2)OCC)cc(N2CCCCC2)ncn1 c1(N2CCC(CSC)CC2)ccc(F)cc1S(=O)(=O)C(F)(F)F Cc1c(C(N2CCC(C(C)NC(c3cccnc3)=O)C2)=O)c(C(F)(F)F)nn1C C1(CCNC(Cc2ccc(CCC)cc2)=O)CN(C(=O)CCOC(C)=O)CC(C)O1 C(=O)(CC(C)c1ccco1)NC(C1(O)CN(C(c2nncn2C)C)C1)C N1(C(CC(CNC(c2ccc(Cl)s2)=O)OC)=O)CC2(C1)CN(C)CCO2 CC(C)C(O)C(C)C(=O)N1CCCC1CCC(=O)NCC(c1ccnn1C)O N1(C(C(C(C)C)O)=O)CCCC2CN(C(C3CC4(C3)CC4(F)F)=O)CCC12 CC(C(=O)N(C)CC1(O)CN(C(C2CCC(F)(F)C2)=O)C1)C(F)(F)F N1(C(C2CC3CCC2C3)=O)CCC(CNC(C2(CO)CCCO2)=O)C12CC2 C(=O)(C#CC1CCOC1)NC1CCC(NC(C23OCCC(C)(C2)C3)=O)C1 O=C(CCC(CF)CF)NC(C(=O)Nc1cccc(F)c1O)c1ccco1 C(CCC(=O)NCCNC(C1(C(C)(C)O)CCC1)=O)=CCC=C C1(CNC(c2scc(C)c2C)=O)CC2CCC1N(C(C1(C(C)(F)F)CC1)=O)C2 C1(CCC(=O)NCCC(C)NC(C2(n3nccn3)CC2)=O)CCCN1C CCCCCC(CC)C(=O)N1CCCC1c1cn(-c2nccnc2OC)nn1 c1(CC(N2CCC(C)(c3cn(Cc4cnc(C)[nH]4)nn3)C2)=O)cnc(Cl)c(C)c1 N1(C(c2ccc(C3CC3C)o2)C(=O)NCC=C)CC2(C)CCC2(C)C1 C1(C)(C(N2CCC(NC(c3ccc(N(CC)CC)cc3)=O)C2)=O)CCCS1(=O)=O C1(NC(c2nc(CC)sc2)=O)CCN(C(=O)C=C(C)C(C)(C)C)CC1O C1(c2cn(C)nc2)CCCC(C(=O)Nc2ccsc2C#N)C1 c1(CCCC)nc(-c2coc(-c3csc(C)n3)c2)n(C2CCSCC2)n1 Cn1cc(C(=O)O)c(-n2cc(-c3ccc(C(N4CC(O)C4)=O)cc3)nn2)n1 CCCC(O)C(=O)N1CC(CO)(NC(c2cc(Br)c(Br)s2)=O)C1 C(c1ccc(Cl)cc1)=CCNCC(c1noc(C(C)C)n1)OCC N(C1c2ccccc2CC1NC(C1CC1CF)=O)C(c1cn(CC2CC2)cn1)=O c1(C(N2CCC(C(N(CCCCCSC)CC)=O)CC2)=O)cccc2ncnn12 C(c1ccc(F)c(F)c1)=C(C(=O)NC1CC(CNC(C(CCCOC)C)=O)C1)C C(C(O)(CC)CC)NC(C1C(NC(C=C(CC)CC)=O)CCC1)=O C1(C(=O)NC(CCC=C(C)C)C)CC(O)CN1C(=O)CC1CNC(=O)O1 C1(OC)CN(C(=O)CC(C)c2ccncc2)CC1NC(C1(C)CC(C#N)C1)=O c1(C(C)NC(N(C(CC)C)Cc2ccccc2)=O)cc(F)cc(Br)c1 CC(O)C(C(=O)N1CCCCC1CN(C(=O)CN1CCSCC1)C)N(C)C c1(C(=O)NCC(CC=C)NC(=O)CCC2CC2(Cl)Cl)cc2cccn2c(O)n1 c1(CCC(=O)NCCCN(C(C(C(CC)O)C)=O)C2CC2)cc(F)c(F)c(F)c1 CC1C2CCCCC2CN1C(C1(C)CN(C(=O)CCNC(=O)CO)C1)=O C(=O)(CC(C)(C)CCOC)NC1(CC=C)CCN(C(=O)C(F)C(C)(C)O)C1 c1(C(=O)NCC(CCCC)NC(C2(F)CCS(=O)(=O)C2)=O)ccc(F)c(O)c1 Cc1c(C(=O)NCCOCCOCCNC(=O)C(C)(C)O)ccc2n[nH]cc12 C(=O)(C1SCc2cccnc21)NCC1CCN(C(C2C(C)(C)C2)=O)CC1 c1(SCCC(=O)NC(C)CCNC(c2cncnc2)=O)ccccc1Br c1(OC)ccc(Cl)cc1C(C(=O)C(CC(C)C)n1ccnc1)=O.N1CCCC1CN n1(CCCCO)nc(-c2cccc(C(F)F)n2)nc1-c1n[nH]c(Br)c1Br c12cnc(cn1)CNCc1ccc-2s1.c1cc(C2CCC2)nn1C.C1CC1 C1(C(=O)NCC2CC(NC(c3csc(C(F)F)n3)=O)C2)CCOC1=O N1(C(COCCCC(C)C)=O)CC=C(C(=O)N2CC(C3CCCO3)C2)CC1 N1(C(c2cc(C)oc2)=O)CC(C2CCCN(C(c3c(C)cccc3C)=O)C2)C1 C1(NC(CC2(OCC)CCC2)=O)CCSC12CN(C(=O)Cn1cnccc1=O)C2 N1(C(C2=C(C)CC2)=O)CCN(C(c2ccnn2CC(F)F)=O)C(C2CC2)C1 N1(C(C2(CCCC)CC2)=O)CCC(CN(C)C(c2cnoc2C)=O)C1 C(=O)(C1=Cc2ccc(Cl)cc2OC1)N(C(C)CCNC(=O)C=Cc1cc[nH]c1)C N1(C(C=C(C)Cl)=O)CC(N(C)C(c2ccc(C(N)=O)cn2)=O)C(F)C1 C1(NC(C2(OC(C)=O)CC2)=O)CCC(NC(c2cc(C3CC3)ccn2)=O)CC1 CC1=C(C(=O)NC2CCCC(NC(c3ccc(COC(C)C)cc3)=O)C2)CCO1 CCC(CC(=O)NC(C(=O)Nc1ccccc1C)c1cccs1)OC c1(NC(C(=O)N(CCC(=O)OC)CC#C)=O)cc(C)ccc1SC CP(C)(=O)CCC(=O)NCC1CCCN1C(=O)Cn1ccc(C2CC2)n1 Cc1ccnc(C(=O)NCC2(O)CN(C(=O)CCCNC(c3cccs3)=O)C2)n1 CCC(CC)(CC)C(=O)NC(C)CN(C(=O)C(C)OCCc1ccccc1)CC c1(CC(N2CC(CNC(C(c3ccc(O)cc3)C)=O)C2)=O)ccc(Br)c(O)c1 c1(C(=O)NCC(C)(CO)NC(CCCCC=C)=O)cc2c(C)ccc(F)c2o1 C=C(C)C1OCCC1C(=O)NCC1(C)CCCN(C(=O)CSC)C1 Cc1c(C(=O)NC2CC(CNC(C3(CCO)CC3)=O)C(O)C2)[nH]c2c1CCCC2 C1(NC(C2(CF)CC2)=O)CN(C(C2C(C)(C)C2CN=[N+]=[N-])=O)CC2(CCC2)C1 C(C(C(=O)NC12CC(C1)C2)NC(=O)CC1C=CCCC1)OCC C(=O)(CCS(=O)(=O)Cc1ccccc1)NC1CCN(C(Cc2nnc(C)o2)=O)C1 C1(N(C(C(n2ncc(C)c2)C)=O)C)CCC(NC(=O)C(C2(O)CCCC2)F)CC1 C12(C(N)=O)CCCC1(C(=O)NC(C1CN(CC3CC(F)(CO)C3)CCO1)=O)C2 C1(O)(CNC(C2C(C=C(C)C)C2(C)C)=O)CCCN(C(c2cncnc2)=O)CC1 C12(CNC(c3cc(Cl)ns3)=O)CCC(CC1)N2C(=O)C=Cc1cccnc1 c1(CNC(C(=O)NCc2cnc3c(c2)CCN3)=O)c(F)ccc(F)c1Cl N1(C(c2c(CC)n(C)nc2)=O)CC2(CCN(C(=O)COc3ccsc3Cl)CC2)C1 c1(OC)c(C(N2CCC(CNC(=O)C(C)(C)OC(C)=O)C(C)C2)=O)ccnc1F Cc1ccc(SC(C)C(N2CC(C(C)(C)O)(CNC(C3CC34CC4)=O)C2)=O)cc1 Cc1ccnc(C)c1C(=O)NC1CCCC1CNC(c1cccc(Br)c1F)=O c1(C(=O)NC2C(C)CCN(C(C(OC)OC)=O)C2)[nH]c2ccc(OC)cc2c1C CCC(CC(=O)NCCN(CC(C)O)C(=O)C=Cc1ccccc1Cl)C(F)F Cc1ccc(Br)cc1C(N1C2CCC1C(NC(=O)C1=CCOCC1)C2)=O N1(C(C(C)N(C(C)=O)C)=O)CCN(C(c2nnc(C)s2)=O)CC1C(F)F N1(C(=O)CCn2cc(-c3cc(C(F)(F)F)ccc3Cl)nn2)CCSC2CCC12 C1(CCN(C)C(C2CC(O)C(F)C2)=O)CCN(C(C2(C3CCC3)CC2)=O)CC1 c1(C(=O)NC(C(C(C)C)NC(CCc2cnc(C)o2)=O)C)cc2cnccc2o1 C1(NC(C(C)n2cnnn2)=O)CN(C(=O)CNS(=O)(=O)C2CC2)CC2(CCC2)C1 N1(CCC(=O)NCC2C(NC(C(C)C(C)(F)F)=O)C2)Cc2ccccc2C1 CON(CC1CC1)C(=O)C(CC(C)C)NC(=O)C1CCc2nccn21 C1(CNC(C(C)(N(C)C(c2ccns2)=O)C2CC2)=O)NC(=O)NC1=O N1(C(CN(C(CCN(C)CCO)=O)C)=O)CCCC(C#N)C1 C(CC(C)C)(C(=O)NC(CN=[N+]=[N-])C(=O)NCCC1C=CCC1)OC C1(CC(=O)Nc2cnn(C3CCCC3)c2)CCCC1NC(C1(O)CCOC1)=O CCCCC(CC)CC(=O)NCC(C(=O)NC(c1cccnc1F)C)N(C)C c1(NC2C(CNC(c3noc(CC)c3C)=O)CCCC2)ncc(C#N)cc1Br c1(N2CC(CCF)OCC2)nccc(=NCc2ccncc2C(F)(F)F)[nH]1 c1(NC(C(c2ccccc2)C)C)ccc(C(F)(F)F)c(Cl)c1 C1(C(=O)N(CCNC(=O)CCCn2cccc2)C2CC2)(CC)CCOC1 C1(NC(C=CC(=O)OCC)=O)COC2CN(C(=O)CCS(C)(=O)=O)CC12 C1(C(=O)NC2COC(C)(C)C2)(CC)CCN(C(c2coc(C3CC3)n2)=O)C1 CCCC(C)(CC)C(=O)N1C2CC1CN(C(=O)Cc1ccc(C)s1)C2 c1(CC(N2CCC(C(C)NC(C(C)OC)=O)CC2)=O)cc(Cl)cc(Br)c1 n1(CC)cc(C(=O)NCCn2ccc(CC3CC(C(C)O)C3)c2)cn1 c1(C(=O)NC(c2csnn2)C)coc(CNC(C2(O)CC(CF)C2)=O)n1 C1(C(=O)NCC2C(C)(C)C2)CCCN(Cc2cccn2C)C1 C1(C(=O)NCCc2ncn(C)c2)(NC(=O)CC23CCC(CC2)C3)CCC(C)(C)C1 N(C1CCCc2ccccc21)C(C1(C)CCCCNC1=O)c1nnnn1C1CC1 N1(C(C(CC)Oc2ccccc2Cl)=O)CCC(O)(CNC(=O)CC2(O)CC2)CC1 C1(NC(=O)C(F)=CC2CC2)CN(C(=O)C(O)CC(F)(F)F)CC12CCC2 C1(COC)CN(C(=O)C(C2(O)CCCC2)F)CCN1C(=O)CN(C1CCCC1)C N1(C(=O)NC(F)(F)C(F)(F)F)CC2CC1CN2Cc1ccc(OC(F)(F)F)cc1 c1(C(C(=O)NC2CC(C)CN(C(c3c[nH]nc3F)=O)C2)C)cc2ccccc2o1 C1(O)(CC)CCCN(C(=O)CN(C(C2(CC)CCOC2)=O)C2CC2)C1 c1(N(CC(C)OC)C)ccc(S(=O)(=O)N2CCc3nc(=N)[nH]cc3C2)c(Br)c1 C1(NC(C2CN(C(N)=O)C2)=O)CC(C(N2CCC2C(=O)NC2CC2)=O)CC1O c1(CNC(c2ccc(O)nc2)=O)ccc(O)cc1.C12(O)CN(C1)C(=O)CNC2=O C(CCCCCC(=O)N(C)CC1CCCN1C(C1CN(C2COC2)C1)=O)SC C1(N(C(C2(C(CC)=O)CC2)=O)C)CCC(NC(C2(C)CCCO2)=O)CC1 c1(NCC(C2CCCCC2)NC(C(C=C)O)=O)nc(O)ccc1C(=O)OC N1(C(c2c(C)ccn2C)=O)CC2OCC(NC(C34CCCN(CC3)C4)=O)C2C1 CC1CCN(C(c2cnccn2)=O)CC1CNC(=O)C(=O)Cc1ccc(Cl)cc1 Cc1cc2c(Br)ccc(C(N3CCCC4C3CCN4C(C3CC3C)=O)=O)c2o1 N1(C(C(CC)=O)=O)CC2CCN(C(=O)NC3CC3C3CC3)CCC2C1 CCCC(O)C(=O)N1CCN(C2CCN(C(c3cc(C)oc3C)=O)C2)CC1 Cc1cc(C(N2CC(CNC(c3cc(=O)n(C)o3)=O)CC2C)=O)c(C)cc1Cl CCC(C(=O)NCCOCCNC(c1c[nH]nc1COC)=O)OC C(C(CC)(CC)C(=O)N(CC(c1nn[nH]n1)C)C)NC(C1C(C(=O)OC)C1)=O C1(c2n(-c3ccc(CC)cc3)nnn2)(NCC=CCSC)CCC(C)(O)CC1 N1(C(C)=O)CCN(C(=O)CCC2CC2(C)C)C(C(c2cnc(Cl)s2)C)C1 c1(C(N2CC(C)(C(N3CC(C(C)(C)C)C3)=O)C2)=O)ccc(N)cc1 Cn1cccc(C(=O)NC2CCCC(NC(=O)CN3CCOCC3=O)C2)c1=O Cn1nc(CNC2CCCN(Cc3cccs3)C2)c(-c2nn[nH]n2)c1Cl C=CCCC(C(=O)OC)NC(C1(NC(c2cc(O)cc(=O)o2)=O)CCC1)=O c1(CNC(c2ccc(C(=O)NCCCOCC)cc2)C)ccc(F)cc1OC C1(NC(C(C)NC(CC)(C)C)=O)CN(C(c2nc(C)oc2C)=O)CC1C N1(C(=O)C2=CCC2)CCC(F)(CNC(C2(CC3CCCC3)CCOCC2)=O)CC1 N1(C(C(C=C)(F)F)=O)CC(CNC(=O)CC2CCN(C)C2=O)OC2(CCC2)C1 C(=O)(C(CC(C)C)C(C)C)NC(C(=O)NC1CC(C=C)C1)COC N1(C(CC2CCC(=O)O2)=O)CCN(C(c2ccc(CO)nc2)=O)C2CCCC12 c1(C(N2C(CN(C(c3c(C)n[nH]c3)=O)C)CCC2)=O)oc(Br)nc1C N1(C(C2N(C(C3N(C)CC(F)C3)=O)CCOC2)=O)CCC(CO)=C(F)C1 C(CCN(C)C)(C(=O)N1CCCC1CC1CCC1)NC(C1CC(C)C1)=O C(=O)(C(O)C(CCC)N(c1ccnn1CCC(F)(F)F)CC)NCCSCC C(=O)(CCC(=O)C(C)(C)C)NCC(C(C)C)C(=O)NC1(C)CCOCC1 CCCCCCCCC(=O)NCC(CCCC)NC(=O)C#CC1CCOC1 C1(C(=O)NCc2ccc(C(=O)NCCn3c(C)cnn3)o2)CCCOCC1 Cc1ccn2cc(C(=O)NC3CC(CNC(C4CCCC(O)C4)=O)C3)nc2c1 N1(C(C=CC2N(C)CCC2)=O)CCC(C)(C)C1CNC(=O)CCCOC(C)(C)C c1(C(C(N2C3C(NC(c4ccncc4O)=O)C(C3)C2)=O)(F)F)cnc(O)nc1O C1(NC(c2cnon2)=O)CN(Cc2ccc(C(=O)O)cc2)CC1F c1(CCNCC(C)Oc2ccccc2)cncc(F)c1 CC(CN(C)C)CCC(=O)N(CCCCCC(=O)NC1(C2CC2)CC1)C CCCC(CCCNC(=O)C1=NOCC1)NC(c1c(C)[nH][nH]c1=N)=O C1(CN(C)C(C2(C)CC=CC2)=O)CN(C(=O)CC2CCC2)CCO1 c1(N2CCC(COc3ccc(C)c(C)c3)C2)nc2ccccn2n1 N1(CC(=O)N(C2CCCCC2)CC)C2CCCC1CN(C(C1CCCN1C)=O)C2 c1(-c2cn(C3CC(C(=O)NCC4C(C(=O)OC)CCC4)C3)nn2)cc(Cl)ccc1Cl C1(OC)(CNC(=O)Cc2cnsc2)CCN(C(c2csc(Cl)c2Cl)=O)C1 N1(C(C2CC(C)NC(=O)C2)=O)CC2CCC(C1)N2C(C1(CF)CC(F)(F)C1)=O C1(C(N2CCN(C(C(C(C)O)C)=O)C(C)C2)=O)CCC(N=[N+]=[N-])CC1 C(=O)(CCC(C)C)NCC(CC=C)NC(=O)CNC(c1cccc(F)c1)=O C1(NC(C2(COC)C=CCC2)=O)CN(C(C2(O)CCC2)=O)CC1C1CC1 C1(C(=O)NCC)N(C(C2CC(F)CN2C(=O)OC(C)(C)C)=O)CC1(C)C CC1CC(NC(c2cnc(C(C)(C)C)o2)=O)CN1C(=O)CN(C)C(N)=O c1(N2C3C(NC(C(C=CCCC)O)=O)(CCC3)CC2)nc(Cl)nc2c1CCOC2 CCC(CC)CCC(=O)N1CC2CCC2(CCNC(=O)COCC2CC2)C1 c1(OC)cccc(C(=O)OC)c1OC(C1CCC(C)(N(C)C)C1)=O CCCCC(CC)C(=O)N1CCN(C(c2ccccc2C(C)(C)C)=O)CC12CC2 c1(C(=O)NCCSCc2cn(CC(C)C)nn2)c[nH]c2c(F)cccc12 Cc1cnc2n1C(C(=O)N(C)CCNC(=O)Cc1cn3c(n1)CCCC3)CCC2 N1(C(CC2C(CC)C2)=O)CCC2(CC1)CC2C(=O)NCCS(=O)(=O)CC c1(C(N(CCNC(=O)CCc2ccncn2)CC)=O)cc2n(n1)CCCCC2=O C1(NC(=O)NCc2ccncc2OC2CCCC2)CC12CCCCC2 CCC(CC)N=C(NC1CC12CCC2)N1CCS(=O)(=O)C2(CCCCC2)C1 N1(C(c2cc(C)ccc2Br)C(=O)NCCCSCC)CCCCC1C1CCCO1 N1(C(C(N)Cc2ncccn2)=O)CC2C(C(=O)O)(C1)CS2(=O)=O c1(C(N2CC(N(C(=O)C=CC3CCC3)C)C(F)C2)=O)ccc(F)c(C(=O)O)c1F C(=O)(CCCCN=[N+]=[N-])NC1C(NC(C(n2ccc(C)n2)C)=O)CCC1 c1(NCCC2=CCN(C)CC2)cc(S(=O)(=O)NCCC2CC(F)C2)ccc1C#N N1(C(CNC(COC)=O)=O)CCCCN(C)CC1.C1CC(=O)N1CC(C)C c1(C(N2CC(CCC)C2)=O)nc(-c2cncs2)nn1C.C(C)(C)(C)O c1(C(C(=O)NCc2cccs2)O)ccccc1OC1(CC(=O)O)CC(C(F)F)C1 c1(C(N(C)CC2CCCN(C(C3CCNC3=O)=O)C2)=O)coc2c1CS(=O)(=O)C2 N1(C(CCn2ccc(C)n2)=O)CCCC(N(C(=O)CC2CCCC2O)C)C1 c1(C(=O)NCCN(CCOC)C(c2cnc(C(C)C)nc2)=O)cnccc1Cl N#CCCCCCC(=O)N1CCOC(CCNC(c2cc3c([nH]2)CCCC3)=O)C1 c1(CC)[nH]c(C(=O)NCC2(NC(c3cncc(C(F)(F)F)c3)=O)CCC2)nc1Cl c1(C(=O)NCCCCCN(C(C(Br)=C(C)C)=O)C)cn(C)c2ccccc12 c1(C(=O)NC2CC(NC(Cc3nc(C)sc3)=O)C23CCC3)coc(S(C)(=O)=O)c1 C(=O)(C1Cc2ccc(Cl)cc21)NCC1(C)CCCN(C(=O)CSCC#N)C1 Cc1cc(C)nc(CNC(C2(NC(C3CCCCCCC3)=O)CCCC2C)=O)n1 C(CCC(=O)NCCNC(=O)C(N1CCCC1)C1CC1)=CC(C)C C(C(C(=O)N(CC(O)CN(C)C)C)NC(=O)C(F)n1ccnc1)OCC Cn1cnc2cc(C(=O)NC3C4CC(NC(C5CCOC5)=O)CC34)ccc12 Cc1nn(C)cc1C(=O)NCc1cccc(CNC(C2OCCOC2C)=O)c1 c1(C(N2CCC(N(C(c3cn(C4CCOC4)nn3)=O)CC)C2)=O)cnc(Cl)n1C C(=O)(C1CCN(C(N2CCSC2c2ccccc2)=O)c2ccc(OC)cc21)OC C1(C(=O)NCC2C(C)(C)C2(C)C)CC(O)CCN1C(c1cccc(O)c1F)=O C1(NC(c2ccc(CCC)cc2)=O)(CO)CCN(C(c2nccnc2C)=O)CC1 Nc1cc(C(=O)NCC2CC(F)CN2C(c2sccc2C(F)F)=O)cc(O)c1 c1(CN2CC(CC)N(C(=O)C(C)(C)OC)CC2)cccc2c1CCC2 CC(C)(C#N)CC(=O)N1CCC(C(=O)NCC(c2ccccn2)O)C12CC2 C(CCCC(F)(F)F)NC(C1C=CCN1C(c1cncnc1)=O)=O N1(C(c2occ(C)c2)=O)CCC2CN(C(=O)Cc3ccc(Cl)c(Cl)c3)CC12 c1(C(N(c2cccc(N(C)C)n2)C)=O)cccc(OC(F)F)c1 c1(C(N(CCCNC(c2cccc(CSC)c2)=O)C(C)C)=O)cc(C#N)[nH]c1C C(C(C)(CC(C)C)NC1CCN(C(C)=O)CC1)NC(c1c(OC)cccc1)=O CC(C)(CC#N)C(=O)NC1CCC(Cn2cc(CC3CC(F)(F)C3)nn2)CC1 CCCCC(C(=O)NC(C)C(F)(F)F)NC(C1COCOC1)=O N1(C(c2ccc(C#C)cc2)C(=O)NC2CC2)CCc2sc(C3CC3)cc2C1 c1(C(=O)NC2C(CNC(C3C(CC(C)C)C3)=O)CC2)cccc2sccc12 C(C(=O)NC1CN(C(=O)C2CC2)C1)(C1(C)CC1)NC(c1cn[nH]c1)=O C(=O)(C1CCCn2ccnc21)N(C1CCCCN(C(c2ncn(CC)c2)=O)C1)C C(=O)(C1=C(C)CC(C)(C)CC1)N1C(CNC(C2C(OC)(OC)CC2)=O)CC1 Cc1n[nH]c(C)c1C(C)CC(N1CCC(C)(CNC(c2n[nH]c(=N)[nH]2)=O)C1)=O O=S(=O)(c1ccccc1C(F)(F)F)CN1CCCCC1Cn1cncn1 C12(NC(COCC=C)=O)CC1CN(C(c1cc(F)cs1)=O)C2 N1(C(Cc2ccc(OC)cc2)=O)CCN(C(c2cncc(O)c2)=O)C(CF)C1 C(CC(C)C)(C(=O)N1CCN(C(=O)CN(C)C2CC2)CC1CS(C)(=O)=O)OC c1(OC(N2CC(CC(=O)NC3C(CNC(C(C)C4CC4)=O)C3)C2)=O)ccccc1 OC1CCCc2ccccc2C1NCCc1cc(F)cc(F)c1 Cc1ccc(NC(C2CCCN2C(C2CC3C(C2)C3(F)F)=O)=O)c(O)c1 C1(C(N(CCCCNC(c2c(OC)cncc2)=O)C)=O)(OC)CCC(C)(C)CC1 CC1CC(NC(=O)Cc2nc(C3CC3)cs2)CCN1C(c1cnn(C)n1)=O c1(C(=O)NC2CC(NC(C3(C)CNC(=O)C3)=O)C2)nc2c(Br)cncc2[nH]1 N1(C(c2ccc(OCCC)cc2)C(=O)NCCOC)CCS(=N)(=O)C(C)(C)C1 c1(CC(=O)N(C(C)CNC(c2cccnc2CO)=O)CC)cc2ccccc2o1 C#Cc1ccccc1NC(C1CN(C(c2cccc(F)c2C)=O)CCO1)=O N1(C(c2c(-c3cn(CCCOC)nc3)c[nH]n2)=O)CCC(=O)C(C)C1 N(C1CC(CC)Oc2ccccc21)C(=O)NC1(CCC)CCC1 c1(C(N(C)CC2(O)CCN(C(C3CCCN3C(N)=O)=O)C2)=O)csc2nccn12 C1(C(=O)OC)CC(=O)N(C)C1C(=O)NCCCNC(C1CCS1(=O)=O)=O c1(C(N2CC(NC(C3CC4(CC4)C3)=O)C3C2C3)=O)cc(O)ccc1Br C1(NC(C2N(CC)CC2)=O)CC2(NC(=O)COc3ccc(Cl)cc3)COC1C2 CCC(CC)C(C(=O)NCC(=O)NCC(C)C)OCCOCCOCCO N1(C(c2cnco2)=O)CC2CCN(C(C3(C4CC4)CC3)=O)CC2C1 CC12CC1CCN2c1nnc(CS(C)(=O)=O)n1CCC#N C1(C)(CNC(CS(CC)=O)=O)CCC(NC(c2nn[nH]c2C(=O)OC)=O)CC1 N1(C(c2c(CC)cncc2)=O)CCC(NC(C23CCCC2C3(F)F)=O)C(F)C1 C(CCCCC(=O)NCC1CC(C)(C)CN1C(=O)CC(=O)NC1CC1)OC N1(C(CCCOC)=O)CCC(NC(c2cccnc2C)=O)C(C(C)C)C1 C(C(F)C(=O)NC1CCC(CNC(c2ccn(C)c2)=O)C1)N(CC)CC Cc1cc(C(=O)NCC2CN(C(=O)C(C)OC3CCCC3)CC2C)c(O)c(C)n1 CC1CCN(C(=O)NCC23COC(C(=O)OC(C)(C)C)(C2)C3)CC1CO c1(N2CCC(NC(C(CCC)NC(N)=O)=O)C(F)C2)nc(Cl)nc2ccccc12 N1(C(C2(N(C(C(=Cc3cn[nH]c3)C)=O)C3CC3)CCC2)=O)CCC(N=[N+]=[N-])C1 CCC(C)C(O)C(=O)NCC1CCCN1C(c1cn(C)ccc1=O)=O N(C(=NCCC1CCC1)NCC1CCCS1)C(C)C c1(CCC)cc(C(N2CCN(C(=O)C(C)N(C)C)CC2)=O)c(C)o1 C1(CNC(C2(SC)CC2)=O)(NC(c2cnc(OC)c(C)c2)=O)CCCCC1C c1(CNC2CC(C(N3CCC4CCCCC4C3)=O)C2)c(Cl)ccc([N+](=O)[O-])c1Cl C(C(C)C)(C(O)C(=O)NC(CC(C)C)C(=O)NCCc1csc(C)n1)OC N1(C(CCOCC)=O)CCCC1CCNC(c1csc(C(C)C)n1)=O N1(C(c2ncccn2)=O)CCCC2(CCN(C(C3Cc4ccccc4C3)=O)C2)C1 C1(Cl)(CNC(N(CC(c2ccccc2Br)O)C)=O)CC12CCC2 c1(C(=O)NC2(C)CC(NC(C(C(C)SC)O)=O)C2)ccc2nnc(S)n2c1 CCC(C#N)C(=O)N(CCCNC(=O)Cc1cnn(CC)c1)C c1(C(=O)NC(c2ccc(Br)cc2F)(C)C)cc(Cl)cnc1O C1(C(=O)NCc2cn(CC(=O)NCc3ccc(F)cc3)nn2)CCCC12CC2 N1(C(C2(SC)CCC2)=O)CCN(C(=O)CC(O)C(C)C)C(C(C)C)C1 c1(C(C)(C)C)nc(CNC(C2C=CCN2C(c2cncnc2)=O)=O)cs1 N1(C(C(C)N2CCCC2)=O)CC(C)C(C)(C(=O)NOCc2nc[nH]n2)C1 Cc1cc(N)cnc1C(=O)NCCC1CCCCN1C(=O)CC1CC1(C)C CCCCC(C)C(=O)N(CC(C)(C)C(=O)NC1CCN(C)C(=O)C1)CC C(CN=c1[nH]c(=NCCSCCS(C)=O)[nH]c2cc(OC)ccc12)NCCO C1(C(=O)NCCn2c(C)nnc2)C2CC2CN1C(C1CC1(C)C)=O c1(C(=O)NCC2CCC(NC(C(c3cncnc3)C)=O)C2)c[nH]cc(Cl)c1=O C(CN=c1nc2sccc2c(NC2CC(C)OC(C)C2)[nH]1)c1ccc(CC)cc1 C1(NC(c2c(C)ccnc2)=O)CCN(C(c2cc(Br)n(C)c2)=O)C(C2CC2)C1 c1(CC)nc(=N)[nH]cc1C(N1CCCCC1CCNC(=O)CC1CSCCS1)=O Cc1ccc(C(N2CCC(c3cccc(O)c3)CC2)C(=O)NC2CCC2)c(C)c1 c1(C(N2CCC(C#C)(O)C2)=O)n[nH]c2c1CN(C(=O)C=CC)C2 CC1COCCC1CNC(=O)CCCNC(c1cnc[nH]c1=N)=O c1(C(=O)NC(C)C(C)NC(c2ncccc2CO)=O)cc(Cl)nnc1O N1(C(C)C(N2CCC(C(N3CCOC4CC34)=O)C2)=O)C(=O)CCCC1=O C(=O)(CC(C(C)C)C(C)C)NCCC1(O)CCN(C(c2cnc(SC)s2)=O)C1 c1(C(N2C(C(C)NC(c3cnc(S)[nH]3)=O)CCC2)=O)cncc2c1CCC2 c1(C(=O)NCCNC(C2CCCN(C(=O)C#CC3CC3)C2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 Cc1cnc2n1CCCC2C(=O)NCCN(C(=O)C(S(C)(=O)=O)C1CC1)C(C)C C1(C2CCN(C(c3cc(C4CCC4)n[nH]3)=O)C2)(NC(=O)C(O)C2CC2)CC1 N1(C(c2n(C=C)ncc2)=O)CCC(C(=O)Nc2ccccc2CC)(CC)CC1 C1(N(C(CNS(NC)(=O)=O)=O)C)CCCCN(C(C2CCC(C)(C)O2)=O)C1 C=CC(C)(O)C(=O)N(CC(C)CNC(c1cnn(CC)c1Br)=O)C C1(CC=C)(NC(=O)C=C2CCCCC2(C)C)CCN(C(=O)C2=NOCC2)CC1 Cc1ccc(NC(c2n[nH]c(C)c2Cl)c2nnnn2C(C)(C)C)c(C)n1 C(=O)(CC1=NNC(=O)C1)N1C(C)C(NC(C2CC3C(C2)C3(F)F)=O)CC1 c1(CC)cccc(C(=O)NC(C)C(C)C(=O)N(C)Cc2cn(C)nc2C)c1 c1(-n2cc(C(=O)NC3CC(CCNC(CC)=O)C3)nc2)cc(C)ccc1OC C1(C(=O)NC2(C)CSC2)CCCCC1CNC(c1sccc1CO)=O c1(OC)ccc(C(N2CC3(C(N4CCCC4C)=O)CC2CO3)=O)cc1OC(F)F C1(C(=O)NC(C(C)NC(CC(C)C)=O)CO)CC=CCC1Cc1ccccc1 c1(CNC2CCCC(P(C)(C)=O)C2)cc(Br)cc2c1OCCC2 C(=O)(C1=NOC(CNC(C2CC3(CCC3)C2)=O)C1)NC(CC#C)CC#C c1(C(=O)NC2CCC(NC(c3nc(OCC)oc3)=O)CC2)cc(F)cc(Cl)c1O Cc1cncc2cc(C(=O)NCC(C)(O)CNC(C3CCSC3)=O)sc12 CC1CC2CC2CC1C(N1CCN(C)C(CNC(c2cc(Cl)c(Cl)n2C)=O)C1)=O C#CCC(C)(C)C(=O)NC(C)CC(C)NC(=O)C(F)C(C)C C#CCC(C(=O)N1CCC(C(C)C(=O)N(C)CCc2ccccc2)CC1)C1CC1 c1(O)ccccc1C.n1(CCCSCCCC)cc(CCN2CCCCC2)nn1 N1(C(c2c(CC)sc(=N)[nH]2)=O)CC(NC(=O)C2=C(C)OCCC2)C2CCCCC12 C(=O)(C(C)(CO)NC(c1cc(OC)cnn1)=O)N1C(CCC=C)CCC1 N1(C(COCCC)=O)CC2CC1CN(C(c1cn(C)nc1C(F)(F)F)=O)C2 C1(C(=O)NCc2c(C)cncc2)CC12CCN(C(c1cccnc1)=O)CC2 c1(C(N2CCC(C(C)(C)C)(CNC(C(C)(C)F)=O)C2)=O)cc2cccnc2s1 C1(C(C)(C)C)(CNC(c2cnc(C)[nH]2)=O)CCN(C(=O)C(C)C#N)C1 c1(C(C(C(C2CCCC2)N)=O)=O)ccnn1C1CC1.C(CN)NC(=O)C1CC1 c1(CCOC)cc(N)ccc1NC(=O)C(C)(C)n1cncn1 C12(NC(C(C)OCCN(C)C)=O)CC(CN1C(=O)CCC(=O)C1CC1)C2 c1(C(=O)NCC2N(C(c3cn(C)c(Br)c3)=O)CCC2)nnc2n1CCCC2 C(CN=c1nc(NC2CCCC2O)c2c(F)cccc2[nH]1)(N(CC)CC)C1CC1 c1(C(=O)NCC2CCN(C(C3CN(S(N)(=O)=O)C3)=O)C2)cnnc2ccccc12 C=CCN=c1[nH]c(C(N2CCC(NC(C3(S(N)(=O)=O)CCC3)=O)C(C)C2)=O)cs1 C1(N(C(C2CCC3CC23)=O)CC)CCN(C(c2ccc(F)s2)=O)CC1 CCCCC(C(=O)NCc1cnc(OC)s1)NC(=O)C(CC1CCC1)OC CC1(CNC(c2ccccc2CO)=O)CCN(C(=O)C(O)Cc2ccccn2)C1 n1(CCCNC(c2cnn(CC)n2)=O)nc2ccccn2c1=O c1(C(F)(F)NC(=O)C(F)CC2CN(C(F)(F)Cl)C2)ccc(N2CCOCC2)cn1 c1(N2CCC(CCNC(CCSC)=O)CC2)nc2ncc(Cl)cc2o1 N1(C(c2c(C)snc2)=O)CCC(C(=O)NCCC(O)CO)CC1C Cc1noc2nc(C(=O)NCCOCCN(C(=O)CN3CC(C)C3)C(C)C)ccc12 c1(OC)ccc(OCC(=O)NCC2(F)CCN(C(C3(F)CCOCC3)=O)C2)cc1 CC(C(=O)NC1CCCC(NC(=O)CCc2cccnc2Cl)C1)C(C)O c1(Nc2ccc(C(N3CCN(CCCC)CC3)=O)cn2)cc(O)c(O)cc1O C=CCCC(C(=O)NCc1cccc(F)c1C)NC(=O)CC1CNC(=O)O1 C1(C(=O)NC(CCSC)C(=O)NCCc2ncc(C)cn2)CC2CC(=O)C1C2 C1(C(=O)Nc2cc(C(=O)OC)c(F)cc2C)CCCC(F)(F)CN1 N1(C(c2ncn(C)n2)C(=O)Nc2c(OC)cccc2)CC(OC)CCC1C N1(C(c2c[nH]c(=NC)o2)=O)CCCC(O)(CNC(=O)C(C)c2cccs2)CC1 CCC(O)C(=O)N1CC(O)(C(C)NC(=O)CNS(=O)(=O)C2CC2)C1 CC1CCCC(CNC(=O)NCC2CC3(CC3)C2)C1 c1(NC(=O)OC(C)(C)C)cnc2n1CCC(C(=O)Nc1cn(CC(F)F)cn1)C2 Cc1cc(C(N2CC(C)(C)CC2CNC(C2CCC(C)(F)CC2)=O)=O)cc(N)c1 c1(C(=O)NC2CN(C(c3cnc(C)[nH]3)=O)C(C)C2)cccc(Cl)c1O C#CCCCCCNC(=O)C(C(C)C)NC(=O)C(C)n1cncn1 C12(C(=O)NCCN3CCN(C(C4CCCC4)=O)CC3)CC=CCN1CCC2 N1(Cc2c(OC)cc(Cl)cc2)Cc2[nH][nH]c(=NC(=O)c3nccs3)c2C1 N1(C(Cn2ccc(C)n2)=O)CC(NC(=O)Cc2cn(C)nc2C)C(C)C1 N1(C(c2c(CC)cns2)=O)CC(CC(=O)NCc2c(C)coc2C)CC1(C)C N1(C(=O)Nc2c(C)ocn2)CC2(CC(C)CO2)C1 C(=O)(C(C(C)C)N(C)C)NCC(CNC(C1(C(=O)OCC)CC=CC1)=O)F C1(C(N2CC(NC(=O)CCF)C(F)CC2)=O)CCn2ccnc2C1 c1(C(N2CC(NC(CC3(CC)CC3)=O)CC2(C)COC)=O)cccc2nsnc12 C1(C2CCN(C(C3CCCCC3(F)F)=O)C2)(NC(c2cn(C)c(O)n2)=O)CC1 C=C(C)CC(C(=O)NC1CN(CC)CC1C)NC(c1cc(O)ncc1F)=O C12(CCCCC1)C(=O)N2.C1(CNC(C(C)C#N)=O)(CO)CC12CCC2 C(=O)(C(CC(F)F)N(C)C(C1CC(O)(C(C)C)C1)=O)NC(CCOC)C(C)C C1(CC(=O)NC2CC(NC(c3sccc3C3CC3)=O)C2)CCCC2(CCC2)O1 N1(CCOCCO)CCC(NC(c2ccc(Cl)cc2)C2CCCNC2)CC1 C#Cc1cc(F)c(C(=O)NC(C)C(CO)NC(=O)CC(C)CC(C)(C)C)cc1F c1(SC)cn(C)nc1C(=O)NC(CNC(C1CCC=CCC1)=O)C(C)(C)C C1(NC(C=C2CCC(C)C2)=O)CN(C(c2cocn2)=O)CCC1C(F)(F)F N1(C(CCc2c(C)noc2Cl)=O)CCN(C(c2csc(C)c2N)=O)CC1C N1(C(c2cnn(C)c2F)=O)CCOCC(NC(=O)CC2CCCC(=O)N2)C1 N1(C(C2CCC(C)(C)C2)=O)CCOCC(F)(CNC(=O)C=CCO)C1 N1(CC(=O)NCCCOC)CCC(NC(C2(c3ccccc3)CC2(C)C)=O)CC1 C1(C2(O)CN(C(=O)COc3ccc(CO)cc3)C2)(CNC(C(CC)C)=O)CC1 CC1CN(C(=O)C(C)(C)n2cc(-c3cncs3)nn2)CC1NC(=O)NC(C)(C)C c1(C(=O)NCC(C)(C)CNC(C2CC2(C)Br)=O)cccc2c1OCO2 CCCC(C)(C)C(=O)NC1CN(C(=O)CCc2ccc(OCC)cc2)CCC1O c1(C(=O)NC(CCNC(c2n(C)ccc2)=O)(C)C)ncc(Br)cc1O N1(C(c2c(C)nn[nH]2)=O)CCC(CNC(c2cccc(C(N)=O)c2)=O)C(F)(F)C1 C1(NC(C(CCOC)C)=O)CCN(C(c2sc(C)nc2C)=O)CCC1(F)F c1(C(=O)NCCCC(C)NC(=O)C(C)N(CC(F)(F)F)C)ncccc1Cl Cc1ccn2ncc(C(N3CC4CCC(NC(=O)CC5(C)CC5)CC4C3)=O)c2c1 C12(C(=O)NCCCN(C(C(COC)(C)C)=O)C)CCCCC1CCC2 c1(C(N2C(CC(=O)NC(C(=O)OCC)C3CC3)CC(F)C2)=O)nc(C)ccc1C N1(C(CN(c2ccc(C)c(C)c2)C(C)=O)=O)CCN(C(CN(C)C)=O)CCC1C C1(CCC(=O)N(CCCCNC(=O)CC2C=CCCC2)C)CCC(=O)NC1 c1(SC)cscc1C(=O)N(CCCN(C(=O)C(C)OC(C)(C)C)C)C Cc1nc(C(=O)NCC2(c3ccccc3)CC(NC(C3CC3Cl)=O)C2)sc1C C1(CNC(CC(CC)OC)=O)CCN(C(=O)CC(C)(C)OC)C1(C)C c1(CC)nc[nH]c1C(=O)N(CCNC(c1scnc1Cl)=O)CCOC c1(C(N2C(CNC(=O)COC(F)(F)F)CCC2)=O)c(Br)ccc2c1OCO2 N1(C(C=CCCC)=O)CCN(C(=O)Cn2nc(C(F)F)cc2C)C2CC12 c1(C(CNC(=O)CCCC2CCC2)NC(C2(C#C)CCC2)=O)ccc(F)cc1F C1(NC(CC2C(CNC(C(C)C3CC3)=O)C2)=O)C=CC(C(N)=O)C1 c1(C(N2CCCC(CCNC(=O)CNc3ncccn3)C2)=O)cc(Cl)cc(Cl)c1 N1(C(C2C=CC(Nc3ncccn3)C2)=O)CCC(CNc2cocn2)CC1 c1(CC)ccc(C(C)C(N2CCCC2CN(C)C(C2CC(O)C2)=O)=O)cc1 C1(CC(=O)N(C2CCN(C(c3ccc(Cl)cc3)=O)C2)CC)CCC(C(C)C)CC1 C(c1cnc(OC)nc1)=CC(=O)NCCN(CCC)C(c1ccc(N)cc1)=O c1(CC)c(C(N2CCC(C)C2CNC(=O)CCc2nc(C)c(C)[nH]2)=O)ccn1C N1(C(C(c2ccccc2C)OCC)=O)CCCC(c2nc(C)c(C)s2)C1 C(=O)(C1=C(C)CCCC1(C)C)NC(C(C)NC(C1(C=C)CCC1)=O)C(C)C C(=O)(C(CNC(C1CC2(CCC2)CO1)=O)C(C)(C)C)N1CC(OC)(CO)C1 n1(CCC(=O)NCC2CCCN(C(c3csc(C4CC4)n3)=O)C2)cnccc1=O C12(C(N(CC(C)NC(=O)CSCc3ccncc3)C)=O)CCCC1C2 C1(C(N2C(CN(C(c3ccc(C)cc3F)=O)CC)CCC2)=O)CCN(OC)CC1 C(=O)(C1=CCC2(COC2)OC1)N1CC(C)C(NC(=O)Cc2cccs2)CC1 CC(CN=C(NC1CCC1)N1CCC(CC(F)(F)F)C1)N1CCOCC1 c1(OC)cnc(C(=O)NCC23CC2CN(C(=O)CC(O)c2ccccc2)C3)cn1 Cc1nc2ncnn2c(N2CC3(CN(C(=O)CC4CCS(=O)(=O)C4)C3)C2)c1C C(C(C)C)(C(O)C(=O)N(CC(C)(C)C(=O)N1CC2CCC2C1)C)OC CC1(C(N2CC(NC(C3CC3c3cn[nH]c3)=O)C2)=O)CCCCC1(F)F N1(C(CN(C(=O)CCC=C(C)C=C)CCOCC#C)=O)CC(C)(C)C1C1CC1 N(C(=NCCc1ccccc1)NC1CCC1)CC(=C1CCOCC1)F c1(C(=O)NC2C(CO)CCN(C(c3n(C)c(S)nc3)=O)C2)ccc2c(c1)OCC2 N1(C(=O)NCC(C2CCCCC2)OC)CCCN(c2ccc(C)cc2)CC1 c1(NC)ccccc1C(N1CCC(C(C)NC(=O)C(F)(F)CN(C)C)CC1)=O C1(NC(c2c(C(C)C)n[nH]c2)=O)CCC(C)(CNC(=O)Cc2nnc(O)s2)C1 c1(CC(=O)NC2C3CCN(C(=O)CC4CCSCC4)C23)ccc(O)nc1 CCCC(C(=O)NC1CC2(C1)CC2N(C(=O)CC(=O)N)C)NC(C)=O.C(C)(C)(C)O N1(C(=O)NCC2C(CC#C)CCC2)CCCC(C(=O)OC)C1.c12nccc(n1)N2 CC1CN(C)CC(C(=O)NCC(=O)NCC2(O)CC2)O1 C1(CC(=O)N(C(CC(=O)N(C(C(=O)OCC)CO)CC)C2CC2)C)CCC(=O)CC1 c1(C(=O)NCC2N(C(COCCCOC)=O)CCC2(C)C)ccc([N+](=O)[O-])n1C N1(C(C2ON=C(C)C2)=O)CC(F)(F)CC1(C)CNC(C1CC(=O)N(C2CC2)C1)=O c1(CC)cc(=NC(=O)C(=O)NCc2ccc(OCC#N)cc2)[nH]o1 c1(NC23CC(C(=O)NCc4n(C)cnc4)(C2)C3)ccc(OC(F)(F)F)cc1 C12(CC(=O)NCC3CC3CNC(c3ncncc3Cl)=O)CCC(CC1)OC2 C1(NC(C(C(CC)O)C)=O)CCC12CCN(C(=O)COC1CCCCCC1)CC2 C(C(=O)NCC1(F)CCN(C(C2CC(C(C)=O)C2)=O)C1)(C(C)C)SCC Cc1ccc(CC(=O)NC2(C3CCCCN3C(c3[nH]cnc3C)=O)CC2)cc1C C(=O)(C(O)C(C)CC)NC(CC)CNC(c1ncccc1OC1CCCCC1)=O C12(NC(C(c3ccccc3)OC)=O)CCCC1N(C(C1CCCCS1)=O)CCC2 C1(CNC(c2c(C)nc(C(C)C)o2)=O)CN(C)CCN1C(=O)C=CC(N)=O c1(C(=O)NCC(CC)NC(=O)CNC(=O)CCC(C)C)nc(O)nc(O)c1OC c1(OC)ccc(CC(=O)N(C)CCN(C(=O)C=C(C)C(C)C)C)cc1 C1(C(=O)OC)CCC(F)CN1C(c1cn(-c2ccc(F)cc2)nn1)=O Cn1ccnc1CCCNC(=O)C(=O)NC(c1nc(CN)no1)C1CCOCC1 c1(C(N2CCC(NC(C(C)OCC=C)=O)(CF)C2)=O)cnc2onc(CC)c2c1 C(CC(C)(C)CNC(=O)COC1(C)CCC1)NC(c1c(C)cno1)=O c1(CN(CCN(C)C)CC)ccc(-c2ccc(C(=O)NCCO)cc2)cc1F CCCC(CNC(C1(CF)CC(=O)C1)=O)C(=O)NCCCn1ccnn1 CCC(CCCC(F)(F)F)N=c1nc2c(cnn2C)c(NC(c2csnn2)C)[nH]1 C(c1cccc([N+](=O)[O-])c1)=CC(=O)NC1(CC)CCCN(C(=O)CS(N)(=O)=O)C1 c1(CC)cc(C(=O)N(CC(C)CNC(c2cc(CN(C)C)on2)=O)C)ccc1Cl C(=O)(CCCCCCNC(=O)C(C)NC(N)=O)NCCC1(COC)CCC1 N1(C(CCCNC(=O)OCC)C(=O)NC(C)CC)CC(C(=O)NC)C(C)(C)C1 c1(C(=O)NCC(CC)NC(c2nnn3c2CCC3)=O)cc(F)cc(Br)c1C C(=O)(C(F)CC(C)(C)NC(=O)Cn1cc(C2CC2)nn1)NC(c1ccns1)C C1(NC(C(=O)NCCN2Cc3ccccc3C2)=O)CCn2nccc2C1 CC(C)CS(=O)(=O)CCC(=O)NCC(C)(C)NC(C1OCCN(C)C1=O)=O N1(C(c2c(CCC)nco2)=O)CCCC(N(C(=O)CCc2c(C)noc2C)C)C1 C(=O)(C(C)(C)C(=O)NCC(c1cccc(Cl)c1)NC(c1sccc1C)=O)OC Cc1cc(COCC(N2CC(C(C)NC(=O)CCCC3CCOCC3)C2)=O)no1 c1(NC(=O)Cc2cnccn2)ccc(NC(c2ccon2)=O)cc1F C(C(CC(F)(F)F)NC(=O)C(F)(F)c1nc(C)cs1)NC(C1C(C(=O)OC)C1)=O c1(COC(C(C)CO)=O)ccc(I)cc1 C1(NC(CCC=CC)=O)CCCCN(C(C2CCN(C3CC3)S2(=O)=O)=O)C1 c1(CC)cc(Cl)ccc1C(=O)NCC1CC(C)(C)CN1C(c1cc(C)c(Cl)s1)=O Cc1nc2c(s1)CCCC2C(=O)N1CCC1CNC(=O)Cn1nnc(=N)[nH]1 C(C(C)(C)CC(=O)NC1CCC(C(N2CCC(C)C2)=O)CC1)OC N1(C(CCc2ccc(=N)[nH]c2)=O)CCC(NC(=O)CCN2CCCC2=O)C(F)C1 C1(C(N(C)C)=O)CC(O)CN1C(=O)NCCF c1(C(N(C(C)CN(C(=O)C(O)P(C)(C)=O)C)C)=O)cccn2ccnc12 c1(OC)ccc(C=CC(=O)NC(C)CNC(=O)CC2CCOC(C(C)C)C2)cc1 C(=O)(C(C)C(C)COC)NCCC1(C(=O)NCCC=CC=C)CCCC1 C(=O)(C1CCCc2cccnc21)NCC1(NC(C(C#N)C2CC2)=O)CC1 C1(C2CCCN(C(c3cccnn3)=O)C2)(NC(c2ccnc(C(C)C)n2)=O)CC1 C=CCC(CNC(c1[nH]ccc1CC)=O)NC(c1csnc1OC)=O C(=O)(C1=CC2CCCC12)N(CC(C)(C)CNC(=O)CS(C)(=O)=O)CC C1(N(c2ccn(C)n2)C(Cc2cc(C)cc(F)c2)=O)CCC2(CCNC2)CC1 c1(CCC(C)=O)cn(CCCN(C(=O)CCn2ccnc2)C2CC2)nn1 CC(C)C(C(C)NC(C1(CCF)CC1)=O)NC(=O)COCc1cccc(Cl)c1 c1(C(=O)NC(C2CN(C(=O)C(C)C(C)(F)F)C2)C)ccc2c(c1)C(=O)NCC2 C1(C(=O)NCC(CNC(=O)CCC(C)N(C)C)OC)(COC)CCCCC1 Cc1cccc2c(C(N3CCC4(CC3)CC4NC(=O)C(C)(Cl)Cl)=O)csc12 c1(C(C(=O)NC(C2CN(C(=O)CC3CCCC3)C2)C(F)F)(F)F)cc(F)cc(F)c1 C=CCC(C(=O)N1CCC(C(C)C(N2CC3(CCCN3C)C2)=O)CC1)C(C)C C(C(=O)N1CC2CCC2(OC)C1)(C(C)(C)C)n1cc(CC(OC)OC)nn1 N1(C(Cn2nc(C)c(Br)c2)=O)CCC2C(C1)CN2C(=O)CCn1ccnc1 C(=O)(C(F)(F)C(C)O)N(CCCN(C(c1c(C(=O)OC)cn(C)n1)=O)C)C n1(C(C)C)ccc(CC(=O)NCC(O)CCNC(=O)COC2CCC2)n1 N1(C(c2ncn(C)c2)=O)CCCC(C(=O)Nc2ccc(C#N)s2)C1 N1(C(C=CC)=O)CCC2(CCN(C(c3cccnc3C3CCNCC3)=O)C2)C1 C1(NC(C(c2ccc(F)cc2)C)=O)CC2CC1N(C(=O)Cn1ncccc1=O)C2 C1(C(N2CCCCC(CNC(C(C(C)C)(C)C)=O)C2)=O)CC12CCS(=O)(=O)CC2 C1(COC)CN(c2cc(NCCc3ncccc3F)ncn2)CC(C)O1 C(C)(C)(CCCC(=O)N(C1CCC1)C)NC(CCCOCCC)=O N=c1nc(O)c(C(=O)NCC2CCC(NC(=O)CN3CCCCCC3)C2)c[nH]1 C1(CNC(CCCOC)=O)CCN(C(C23CC(CN2C2CC2)C3)=O)C1(C)C N(C(=NCCCSC)NC(c1ccc(Br)cc1)C)CC(C)(C)OC C=C(C)CC(C)C(=O)NCCNC(C1CN(C(=O)OC(C)(C)C)CC12CC2)=O C(c1cccnc1C)=CC(=O)NC1CCN(C(C(C)SCCCC)=O)CC1 Cc1nn(C)c2nc(C(N3CCC(C)N(C(C4CC4CF)=O)CC3)=O)ccc12 C1(C(N2CC(CCNC(C(=Cc3ccccn3)C)=O)C2)=O)CCS(=O)(=O)N1C Cc1ccc(C(N2CC3CC3(CNC(c3sc(Br)nc3C)=O)C2)=O)cc1 c1(C(=O)NCC(CNC(c2ccc(OC)cc2Cl)=O)(C)O)n[nH]c2c1CCCC2 N1(C(c2c(C)cc(C(F)F)o2)=O)C2CCCC1CN(C(c1cnco1)=O)C2 c1(C(N2CC3C(N(C(=O)CC4CSC4)C)C3C2)=O)ccc2nnn(C)c(=O)c2c1 C(=O)(CC(F)(F)C(F)(F)F)N1CC(CC=C)(C(=O)O)C1 C(=O)(C(CC(C)(C)C)OC)NCC1CN(C(C(C)NC(=O)NC)=O)CC1O c1(C(=O)NCC2(NC(CCC(C)(C)F)=O)CCC2)n[nH]c2cc(Br)ccc12 c1(C(N(C2COC(C)C2)CC)=O)ccc(CNC(=O)C2CC2)nc1 c1(CCC(=O)N(CCOC)CCNC(C2(O)COC2)=O)cccnc1Cl C(=O)(CCC(=O)NN(C)C)NC(C1CN(C(c2cc(C(C)=O)oc2)=O)C1)C CC(CNC(C12CC(C#N)(C1)C2)=O)C(F)C(=O)N(C)CCOC(F)F N1(c2ncc(C(=O)OCC)s2)CCCC2CN(C(=O)CCSC)CCC12 c1(CC(N2CCOC(c3cn(C4COCC4O)nn3)C2)=O)cnc2ccccn12 C(CNC(=O)C(C)(F)F)(C(=O)NC(CC1CCCC1)CO)N(C)C C(N=c1cc(C)[nH]c(=NC(C)CC(C)(C)C)[nH]1)c1c(Cc2c(OC)cccc2)cccc1 c1(C(=O)NC(C)CNC(=O)CN(C2CCSC2)C)ccc(F)c(C(F)(F)F)c1 c1(OC)cc(C(N2CCOCC2CC(=O)NC2CCC(F)(F)C2)=O)cc(Cl)n1 C1(=O)C(C)NCCN1.C12(C(N(CC(=O)NC(=O)NC)C)=O)CC(C1)C2 C1(NC(C=CC=CCC)=O)CCN(C(=O)CC2(CSC)CC2)C(C)C1 C1(F)(CNC(C2CC(=C)C2)=O)CCC(NC(=O)C(c2ccc(C)cn2)(F)F)C1 CC(O)(C(=O)NCCCOCCNC(c1cn(CC(N)=O)nn1)=O)C1CCC1 C(=O)(N=c1[nH]cc(C#N)cc1C)Nc1cc2cc(C)c(Cl)cc2[nH]1 c1(C(N2CCC(CNC(=O)C(F)(F)F)C2)C(=O)NCC=C)cccc(Cl)n1 c1(C(=O)NCC2(C(F)F)CCN(C(CCC#CC)=O)C2)cnc(OC)c(C)c1 Cc1cc(C)n2ncc(C(=O)NC(C)CNC(=O)C(O)c3ccco3)c2n1 C1(C(=O)OC)(OCC(CNC(C)C)(C)C)CC(C)C1 n1(CC)ncc(S(=O)(=O)NC2(c3ccc(F)cc3)CCCC2)c1Cl C1(CC(=O)NC(CC2CCC2)C(=O)NCc2cn[nH]c2)CCCOCC1 C1(N2CC(CO)C2)CCN(N2CCn3c(Br)cnc3C2)CC1 c1(CC)noc(CC)c1CC(=O)NC(C)C(C(C)C)NC(=O)CC(F)(F)F N1(C(COc2c(C)cc(C)cc2C)=O)CCC2(CCCN(C(=O)C(N)=O)C2)CC1 C(C1CCc2nccn21)NC(C1C2C(NC(=O)CCOC3CCC3)C3C(C2)C31)=O C1(NC(C2(CCNC(CCCOCC)=O)CCCC2)=O)CCC2CC2CC1 C(=O)(C(C)(C)C(C)(C)O)NCCC1N(C(CC(CC)C2CC2)=O)CCCC1 C1(C(N2C(C(C)NC(=O)CCN(C3CCCC3)C(N)=O)CCC2)=O)CCN(C)C1=O C12(C(=O)NCC(CC)NC(=O)C(F)(F)C(C)O)CCCCN1CCC2 c1(CC)ccc(N2CCC(CNC(=O)C=CCN(C)C)C2)c([N+](=O)[O-])c1 N1(C(C2CCCN2CC2CCCO2)=O)CCC(NC(C23CC(C2)C3)=O)CC1 C1(NC(c2cnn(CC(F)F)c2)=O)CCC(CNC(c2cc(Br)c[nH]2)=O)C1 NCC(=O)NNC(=O)C(N1CCOCC1c1ccccc1Cl)c1ccccc1 C1(OC)CC2(CCN(C(C34CC(C)(CN3C(=O)C#CC3CCC3)C4)=O)C2)C1 CC1=C(C(=O)NCC(C(=O)NCC(c2cccs2)O)C(C)C)CCCO1 N1(C(CN2CCC(C)CC2)=O)CCC(NC(C2CCCC(=O)N2C)=O)C(F)C1 c1(C2CCN(C(c3c(OC)scc3)=O)C2)ccc(C)cc1 C1(C(=O)NCC2CN(C(=O)C3=CCCS3)C2)CCc2ncnn2C1 N(C1CCCn2ccnc21)C(C1C(C)(C)CN(C(=O)C(O)CC2CCCC2)CC1)=O c1(CC)ncncc1C(=O)NCC1CC(NC(=O)C=CCCC(C)C)C1 C1(CNC(C2C(C(C)O)C2)=O)CCN(C(=O)C(C)Cc2cnc[nH]2)CC1(F)F N1(C(C2CC(=O)C2)=O)C(C(=O)Nc2ccc(C3CC3)nc2)CCC12CC2 N1(C(c2nc(COC)sc2)=O)CCC2CN(C(=O)C(n3ccnc3C)C)CC12 c1(-n2cc(C(CC)(C)O)nn2)ccc(CCC(=O)NCC2CCS(=O)(=O)C2)cc1 c1(C(=O)NC2C(NC(CC3C(CC)C3)=O)CCC2)ccc(-c2cnc[nH]2)cc1 c1(C(N2CC3(CN(C(Cc4cc(C)no4)=O)C3)C2)=O)cccc2ccc(Br)cc12 C(=O)(C1=NN2CCCN=C2N1)NCC(CNC(C(c1c(C)noc1C)C)=O)O C1(NC(c2c(C)cc(C)nc2)=O)C(CNC(c2csc(CO)n2)=O)CCC12CCC2 c1(NC(C2CC(NC(=O)Cc3cccnc3Cl)C2)=O)ccc(F)c(F)c1 C1(C(=O)OCc2cc(OC)no2)CCN(C(=O)CCC(=O)N2CCOCC2)CC1 C1(OC2CN(C(C)=O)C(CO)C2)CCCC(=O)N1C.C12CCCN1C2=O C=C=CC(C)C(=O)NC1(CCNC(c2cnccc2C(C)(C)C)=O)CCC1 C(C(C)(C)CCNC(=O)C(C)C1CCCO1)NC(C=C(CC)CC)=O C#Cc1ccc(CNC(=O)C(C)N(C(=O)C(C)c2cc[nH]n2)CCC)cc1 N1(c2ncc(CC)cn2)CCCC2(CCN(c3ncc4ccccc4n3)C2)C1 n1(C(CC)C2CCC2)nnnc1C(C)(CSc1ncns1)NCCn1cnnc1 CC1=C(F)CN(C(C2CN(C(=O)CC3(C)CCC3)CC2C(C)C)=O)CC1 C(=O)(CC(C)(C)COC)N(CCN(C(=O)CCC12CCC(CC1)C2)CC)CC C1(CCNC(c2c(CC)oc(C)c2)=O)CCN(C(=O)CC#N)CC1(F)F C1(C(=O)NC2(C)CCN(C(c3n(CC)ccn3)=O)C2)CCc2ncnc(C)c2C1 Cc1ccc(C2CC2)c(CNC(C2CCCN(C(=O)CCC(N)=O)CC2)=O)c1 C1(NC(c2cc(F)c[nH]2)=O)C2CCC(C2)C1C(N1CCC1CO)=O Cc1cn2nnc(CNC3CC3CF)c2c(O)n1 Cc1c(Cl)nc[nH]c1=NCC(O)CNC(=O)NC1CCN1C1CCCC1 Cn1cnc2[nH]c(C(N3CCC(NC(c4ccc(Br)o4)=O)C3(C)C)=O)cc12 N1(C(C(C2CCN(C(CSC)=O)C2)(C)C)=O)CC(C)(C)C1C1CC1 N1(C(=O)CCc2nncs2)CCC2CCC(C1)N2C(C1CC2(C1)CC2F)=O c1(OCC(=O)NCCC(C)(C)NC(=O)CCC2CCC2)cccc(N)c1 C=CCCCCCNC(C1C2CC1N(C(c1cncnc1)=O)C2)=O N1(C(C2(CCC)CCC2)=O)CC2(CCCC2NC(=O)CCCC(C)=O)C1 C1(COC)CCCC2(CN(C(C3(C(=O)OC)CC3)=O)C2)O1.C1CCC(C)C(=O)N1 N1(C(C2C(C)C2)=O)CCCC(NC(c2c(Cl)nsc2Cl)=O)C1 c1(C(=O)NC(CC)CNC(C2CCC(C(N)=O)O2)=O)ccc2nnc(S)n2c1 Cc1cc(NC(=O)C(C)C(C)O)ccc1NC(=O)CCCN=[N+]=[N-] N1(C(C(c2cccc(Cl)n2)CNC(C)=O)=O)CCc2c(CO)cc(Br)cc21 N1(C(c2cccc(OC)c2)=O)CC2CC(CNC(=O)C(N3CCOCC3)C)C2C1 N1(C(C(CSC)O)=O)CCOCC1CNC(c1sc(-c2ncccn2)nc1C)=O C=CCCCCCCC(=O)NC1CC(C)CN(C(c2cnc(S)[nH]2)=O)C1 C(=O)(C(C(C)C)NC(c1ccco1)=O)NCCC1CN(C(C2(C=C)CCC2)=O)C1 N1(C(C2(OC)CC(C)(C)C2)=O)CCCCC(C(=O)NCC(F)(F)C(N)=O)C1 N1(C(COCCOCC#C)=O)CC2CC(C1)N(C(c1cc(=O)n(C)o1)=O)C2 c1(C(=O)NC(C2CCCN2C(C2CCC(=O)O2)=O)C)cn(C)c2ccc(Cl)cc12 C1(C(=O)NCCNC(C)=O)CC(C)CN(C(=O)Cc2nncn2C)C1 n1(CC)ccc(C(=O)N(CC(C)C(=O)NCCC2CCC3CC23)C)c1C C1(C(=O)NC(CCC)C(N)=O)CC1C1CN(C(=O)CC2COCCOC2)C1 CCC(CC)C(C)C(=O)N(C)CC1CCCCN1C(C1CC2(C1)CC2(F)F)=O n1(CC2(CC)CCOCC2)c(-c2ccnn2C)csc1=Nc1ccc(F)c(Cl)c1 Cc1ccc(CC(N2CCN(C(=O)Cc3c(Cl)cnn3C)C3CC23)=O)c(F)c1 C(=O)(C(CC=CC)NC(c1cc(C2CC2)[nH]n1)=O)N(C(C=C)C1CC1)C C12(C(=O)NC3C4CCC5C(C4)CC35)CC(C3CCNCC3)(C1)C2 C(CO)(CC(C)C)NC(C12CC(NC(C(CC)N(C)C)=O)(C1)C2)=O c1(C(=O)NCCC(C)NC(c2c(CCC)nco2)=O)cccc(C(=O)OCC)c1 C(=O)(C#CC1(C)COC1)N(CCCNC(=O)C(C1CCCCC1)F)C C1(CCC(C)C)C(=O)N1.CCC(CCC(=O)OC)NC(=O)COc1cnn(C)c1 CCCCCC(C)CC(=O)NC(C)CCN(C(=O)Cc1coc(C(F)F)n1)C Cc1cn2nnc(C(=O)N(C(C)CCNC(c3nncn3C)=O)C)c2c(O)n1 C1(C(=O)NC(C)CCN(C(=O)COC(C)(C)C(F)(F)F)C)CCCCN(C)C1=O N1(C(=O)NCCC)CCC(C)(C(=O)NC2CCCC2C(N)=O)C1 c1(C(N(C)C)=O)ccccc1C(=O)NCC1CCCCC1NC(C1CC12CC2)=O N1(C(COC(CC)C)=O)CCC(CNC(C23CCCC2C3)=O)(COC)C1 CCCC(C)(O)CC(=O)NCC1CCCCN(C(c2cc(C)ccc2OC)=O)C1 N1(C(c2nnc(C)s2)C(=O)NC(C(=O)OC)C)CCc2c(cc(F)c(F)c2F)C1 c1(OC)cc(C(N2CCCC2C(C)NC(=O)C2=CCOC2)=O)ccc1Br C1(NC(Cc2cncc(C)c2)=O)CCN(C(=O)CC(O)C2CC2)CC1C N(C(=NCc1cn(CC)nn1)NCC1(CC)CCOCC1)C(C=C)C C1(NC(C2C(C)OCC2)=O)CC2CCC(C1)N2C(c1cccc(-n2cncn2)n1)=O N1(C(C23OCC(N)C(C2)C3)=O)CCS(=O)(=O)CC1c1ccc(C(F)(F)F)cc1 Nc1cccc(C(=O)NC(CNC(c2cccc(CO)c2)=O)CC(F)(F)F)c1O C(=O)(C(O)P(C)(C)=O)NCC1(C)CCCC1NC(=O)Cc1ccc(O)nc1 Cc1ccncc1CC(=O)NCc1cnn(C)c1C(=O)NCCc1cncs1 CCCC(C(=O)NC(Cc1cccc(Br)c1)C(=O)O)OCC CN1CCc2nc(C(N3CCC(CN(C(=O)Cc4cnc[nH]4)C)C3)=O)sc2C1 Cn1nc2c(c1C(N1CCCC1CNC(=O)C(O)C(F)F)=O)CCCC2 N(C1CCCc2nccnc21)C(C1CCC(S(C)(=O)=O)C1)=O C12CN(CCC13CN(C(=O)C(n1ccnc1C)C)C3)C2=O.C(=O)(OCC)OC C1(C)(C(=O)OCC)CCN(N2CC(Oc3ccccc3)C2)CC1 C(CCCCCC(=O)NCCc1cn(C)cn1)NC(Cc1ccc(C)cc1)=O Cc1ccccc1CCC(=O)NCC(C(C)C)NC(c1c(C)n[nH]c1C)=O N1(C(C2OCCC(=O)C2)=O)CC(NC(C2CCCO2)=O)CC(F)C1 N1(C(C(C(C)C)=O)=O)CC(C2CCCCN(C(=O)C(C)Cc3ccccc3)C2)C1 N12CC(C(F)(F)C1)C2=O.N1(C(=O)OC(C)(C)C)CCOCC1CNC(=O)C=CCF N1(C(C(C)n2cccn2)=O)CCCN(C(c2cc[nH]c(=N)c2Br)=O)C(C)C1 C(=O)(C(CCN(C)C)NC(c1ccsc1C)=O)NCc1c(COC)noc1 c1(C(N2CCSC2c2ccco2)=O)ccc(O)c(C(=O)O)c1 c1(C(=O)NCC(C)NC(c2cc(CCCO)on2)=O)cnn2c(N)ccnc12 c1(C(=O)NC2CCCC(NC(C3(C(N)=O)CC3)=O)CC2)cc2ncccn2n1 C12(C(N3C4C(NC(C(C)OCCC(C)C)=O)C(C4)C3)=O)CC1COC2(C)C c1(-c2c(C(=O)NC(C)CC3CCCCC3)scc2)ccc(Cl)cc1Cl CC(CC(C)(C)C)C(=O)N1CC2CN(C(=O)C(CO)C(F)(F)F)CC(C1)O2 Cn1cc(C(=O)NCCOC2CCN(C(C3C4CC5C(C4)C35)=O)C2)c(C(F)F)n1 N1(C(C2N(C(CSCC)=O)CCCC2)=O)CC2CC(C)C2C1 C12(CNC(CC(=O)OC)=O)COCC1CN(C(C1CC(OC)CN1C(C)=O)=O)C2 Cc1cc(F)c(C(N2CCN(C(C3CCCCN3C)=O)CC2C)=O)cc1Br C=CCCN=C(NCC1CC(c2ccccc2F)C1)NCC(F)=C(C)C c1(SC)cccnc1C(=O)Oc1ccnn1C.C(=O)(C(C)C)N1C2C(C2)C1=O c1(C(=O)NCC(CC(C)C)NC(C2C(CC)C2)=O)c(C(C)C)cccc1C C1(CN=[N+]=[N-])CCN(C(C2OCCC2NC(=O)CCCF)=O)C1 C1(CNC(c2c(CC)ocn2)=O)CC(NC(=O)C(c2ccncc2C)C)C(O)C1 N1(C(c2c(COC)noc2)=O)CCN(C(c2ncn(C(C)(C)C)n2)=O)CC1 Cc1c(NC(C2(O)CCCC2)=O)cccc1C(c1cc(F)cc(F)c1)=O C1(CSc2cnc(N3CCC(CC)C3)nc2)CCC(Br)C(C(=O)OC)N1 CC(C)C(O)C(=O)NCC1CC1NC(c1ccc(C2CNC(=O)C2)cc1)=O c1(C(N2CC3=C(CN(C(C(C)C(F)F)=O)C3)C2)=O)ccc(C#CC2CC2)cc1 C(=O)(C(C(=O)NCC1CCCN1C(c1ncn(C)n1)=O)C1CC1)OCC CC1(C)Cc2[nH]nc(C(=O)NC3CN(C(=O)CC4CNC(=O)C4)CC3O)c2C1 C(=O)(C(C)(C)CCC(=O)OCC)N1CCC(C(CO)NC(CNC(C)=O)=O)CC1 N1(C(COCC=C)=O)CCCN(C(=O)Cc2cccc(C(N)=O)c2)CC1 C1(C(N2CCC(N(C(=O)C=Cc3cocn3)CC)CC2)=O)CCS(=O)(=O)C1(C)C C1(NC(=O)C(c2cccc(Br)c2)O)C2CCC1CN(c1ncnc3occc13)C2 Cc1c(N)cc(C(N2CC(NC(c3cc(F)c[nH]3)=O)CC2(C)C)=O)cc1[N+](=O)[O-] c1(C(=O)O)cc(CN2CC3C(C(N4CCOCC4C(F)(F)F)=O)C3C2)ccn1 Cc1cc(N2CC(C(C)NC(=O)CN3CCCCC3)C2)cc(C#N)c1[N+](=O)[O-] N1(C(CSCCCC)=O)CC2CC1CCN2C(c1cnccc1Cl)=O n1(CCC)ncc(CNC(=O)C(c2ccc(C)cc2)C)c1Cl C1(C(=O)NCCCCCCOC)CCCCCCN1C(c1occ2c1CCC2)=O CN1CCOCC1C(=O)NCCCN(C(=O)CCc1ccccc1F)CCO c1(C(C)=O)c[nH]c(=NCC(C)CNC(=O)CN2CCc3ccccc32)c(C)c1 CC(C(=O)N(OC(C)(C)C(=O)OC(C)(C)C)OCc1ccccc1)C1CCOCC1 c1(C(=O)NC2CN(C(CCc3onc(CC)n3)=O)CC2C)c(F)ccc(C)c1O C(C(C)C(=O)N(OC)C(C)CCC)NC(CCOCC#C)=O CCCCC(CNC(=O)COC(F)(F)F)NC(=O)CCC(=O)N1CCC(O)CC1 C1(C(=O)NCCCCC(C)NC(c2c(C)snc2)=O)CN=C2N=CNN2C1 n1(CCCOC)nnnc1C(c1cnn(C2CC2)c1)NCc1csc(O)n1 N1(C(C2C(CCOC)C2)=O)CC2CC(C)N(C(=O)CCc3ccccc3)C2C1 C(C(CC(C)C)C(=O)N1C2CCC1CN(C(=O)C(C)=C1CCCC1)C2)OC N(C1CCC(NC(=O)C(=O)C(C)(C)C)c2ccccc21)C(c1scc(C)c1Cl)=O N1(C(=O)CCn2cccn2)CCOC2(CCN(C(C3(O)CC3)=O)C2)C1 c1(C(=O)NCCNC(=O)CC2NC(=O)NC2=O)cccc2ccoc12 C12(NC(=O)C(=O)NC3CC3)CCC(C1)N(C(c1ocnc1C(F)(F)F)=O)C2 C1(c2nn[nH]n2)(NC(C(c2noc(C(C(C)(C)C)N(C)C)n2)C)=O)CCN(C)C1 n1(CC(C)NC(c2cnc(Br)s2)=O)cc(CCCc2ccccc2)nn1 Cn1nnc2c(C(=O)NC3CN(C(=O)CP(C)(C)=O)C4(CCCC4)C3)ccnc12 C(CC1=CCN(C(=O)C(C)=C2CC2)CC1)NC(c1[nH]nc(OC)c1Cl)=O CS(=O)(=O)CCC(=O)NC1CC2CC1N(C(=O)Cc1ccsn1)C2 c1(C(N(C(CNC(CC(=C)Br)=O)C)C)=O)cc(C)c(C)c(S(N)(=O)=O)c1 C(CCCCCC(=O)N1CC2C(C1)C2(C)C)NC(CC(C(=C)C)OCC)=O N1(C(c2cc(C)[nH]n2)=O)CC2OCCN(C(c3cnc4n[nH]c(C)c4c3)=O)C2C1 C(=O)(CC1CCOc2ccccc21)NCC1C(NC(C2C(C)C2C)=O)CCC1 C1(C(C)C)CCC(C(=O)NC2CCC3(CC3)C2)N1C(c1cnc(Cl)n1C)=O c1(NC(C(C=C)C)=O)cccc(C2CC(F)(F)C2)c1 C=C(C)CCC(=O)N1CCC(O)(C(C)NC(C2CCN(c3ccncc3)C2)=O)C1 C1(N(C(C=CCN(C(c2c(C)nsc2)=O)C)=O)CCO)CCCCCC1 c1(OCC)ccc(C(=O)NCC2CC2CNC(=O)C(CN(C)C)C(C)C)cc1Cl c1(C(N(C2CCN(C(C(C)C3CCC3)=O)CC2)CCO)=O)cn2cccnc2n1 c1(CN2CCC(C)(C(N3CCOCC3)=O)C2)cccc2c1OCCO2 C1(C(=O)NC2CC(COC)C2)CCN(C(C2CCCC2O)=O)CCO1 N1(C(C(C)CN(C)C)=O)CC(NC(c2ncn(C)n2)=O)C(c2cncn2C)C1 C1(C)(C(=O)NC(C2C(C(=O)NC3(CC)CC3)C2)C)CCCCO1 CC(CCCCCO)NC(C1(C)C=CCN1C(=O)CC(=O)N(C)C)=O CCC1=NOC(C(=O)NCCCC2(NC(=O)CC3CCCCCO3)CC2)C1 Cc1c(C(=O)NC(CNC(C2CC2C(F)F)=O)C2CC2)cccc1C#N N1(C(C2CN(C(C)=O)C2)=O)CCC(NC(=O)C(C)(C)C2CC2)C1c1ccccc1 Cc1c(C(=O)Nc2cccc(Cl)c2N2CCCCC2)cnc2nncn12 S(=O)(=O)(c1c[nH]ccc1=NC1CCCOC1OC)N(C(CC)C)C CP(C)(=O)CCC(=O)NCC1CCCCCN1C(c1cnn(CCC#N)c1N)=O c1(OC)ccc(CC(=O)N(CCCNC(=O)CC2CN(C)C2)C)c(Cl)c1 C=CC1(C(=O)NCCCc2cnn[nH]2)CCN(C(C2CC(C3CC3)C2)=O)CC1 N1(C(CC2(C=C)CCC2)=O)CC(C)CN(C(=O)C=CI)CC1C c1(C(C)C)c(NC(C2CCN(C(=O)COCC3CC3)CC2)=O)cccc1F CC(O)(C(=O)N(CCNC(c1ccn(C2CCCC2)n1)=O)C1CC1)C1CC1 CC1=CCC(OC(c2nn(-c3ccccc3)nc2C)=O)CC1 N1(C(CCC2OCC(C)(C)C2)=O)CCC(O)(CCNC(c2occc2F)=O)CC1 C(CC(C(=O)N(CC(C)C(C)(C)C)C)NC(=O)Cc1ccccc1O)SC c1(C(N2CC3C(NC(CCSc4n(C)nnn4)=O)(C3)C2)=O)ccn2c1CCCC2 c1(C(=O)NCC2N(C(C(CC)C#N)=O)CCCC2)ccc2cc(OC)ccc2n1 CCC(C)C(C(=O)N1CC(N(C(=O)CCc2nnc(C3CCCC3)o2)C)C1)OC c1(CC)nc(C)c(Cn2cc(C(C)N(C)C(C3(C(C)(F)F)CC3)=O)nn2)o1 Cc1cccn2c(CC(N3CCC4(CCCN4C(C4C(C)C4C)=O)C3)=O)cnc12 c1(C(C(=O)NCC(C)CN(C(=O)CC2CSC2)C)O)ccccc1F C=CCC(C)(C)CC(=O)N(C1CCN(C(C23CC(N=[N+]=[N-])C2C3)=O)C1)CC Cc1ccc(Br)c(NC(=O)C(C)(F)F)c1F.N12CCC(CC1)SCCC2=O C1(CN(C(=O)CCCCC2CC2)C)C2CN(C(=O)COC3CCC3)CC12 C1(O)(CN(C)C(C2CCC(F)(F)C2)=O)CCN(C(c2csc(Cl)c2)=O)C1 C1(NCC(N2CC3C(CNC(c4cc(SC)oc4)=O)C3C2)=O)CCC(F)(F)CC1 c1(CCC)ccc(N)c(C(=O)NCC2CCCC2NC(=O)CC2CC=CC2)c1 c1(C(CCOC)C)nc(C2CCOC2)nn1-c1cncc(Br)c1 C1(NC(CC2CC(C)(C)C2)=O)CC2CC1N(C(=O)CCSC1CCCC1)C2 CC(C)CC(C(=O)N1CCC(NC(c2ccccc2)C2CC2)C1)NC(N)=O Cc1nn2c(C(=O)NCC3COCCN3C(c3cn(C)[nH]c3=N)=O)c(C)nc2s1 c1(C(=O)NCC2(COC)CN(C(c3ncn(CC)c3)=O)C2)c(C)ncn1OC C(C)(CCC(=O)NC1CC(=O)N(C2CN(C(=O)COC)C2)C1)OCC CCS(=O)(=O)c1ccc(Cl)c(C(=O)NCC2CCC2NC(C2CC2C(C)C)=O)c1 C1(CC(=O)N(CC(C)CNC(c2csc(C(N)=O)n2)=O)C)C=NN(C)C1=O N1(C(C2CCC(=C)CC2)=O)CC(OC)CC1(C)CNC(C1CN(C(C)C)C1)=O c1(C(N2CCN(C(c3cn(C)nc3)=O)C3(C2)CC3)=O)cccc([N+](=O)[O-])c1I c1(C(=O)NCC2(OC)CN(C(c3cccn(C)c3=O)=O)C2)nnc(O)cc1O C(=O)(C(CC)CC(C)C)NCCc1c[nH]c(=NCc2c(C#C)cccc2)s1 C(N=c1[nH]c2c(c(=NCCC3CCCO3)[nH]1)CSC2)C1(C)CCC1 c1(C(N2CC(=C(CNC(=O)C=Cc3cncs3)F)C2)=O)nc(Cl)ccc1F Cc1c(C(=O)NC(C)CNC(C2CC3C(C2)C3(F)F)=O)cc(C)c2ncccc12 N1(C(C(=O)NCC2(C(=O)OC(C)(C)C)CCC2)=O)CCOCc2c(Br)cccc21 c1(C(=O)OC)ccccc1OCC(=O)NCCCC(C)(C)NC(=O)CC1CCC1 n1(CC)cc(CCNC(=O)C(CNC(c2nsnc2O)=O)N(C)C)cn1 N1(C(c2cc(CCC)[nH]n2)=O)CC(NC(C2CCCN(CC(F)F)C2)=O)CC1C C1(C(=O)NCc2cn(CC)nc2)CCC2CCC1N2C(=O)CCn1ccnc1C c1(CC(=O)N(CC(C)(C)CNC(=O)Cc2c[nH]nc2C)CC)cnn(C)c1C CCCCCCC(CN(C1CCOCC1)Cc1ccc(C)o1)CC CCCC(CCCNC(=O)CCc1cncs1)NC(c1scnc1CC)=O N1(C(CC(C)(C)OC)=O)CCCC(NC(c2n[nH]c(C)c2Br)=O)C(F)C1 N1(C(c2c(C)cccc2)=O)CCC2(C(N3CC(O)(c4nn[nH]n4)C3)=O)CCCC12 N1(C(C=CCOC)=O)CC2C3CCC(C2C1)N(c1cc(-n2ccnc2)ncn1)C3 c1(C(N2CCC(CNC(C3(C)C(C)CCC3)=O)CC2)=O)ccc2oncc2c1 N1(C(C2CCCC3CC23)=O)CCC2(CCCN2C(=O)C=C2CCC2)C1 Cc1cn(C)nc1C(N1CC(CCNC(c2cc(C(C)(C)C)on2)=O)C1)=O C1(C(=O)NCc2c(C)ncs2)C2CCC(C2)N1C(C1CCCC(C)C1)=O C(C(CC(=O)N(C1CCCC(O)C1)C)NC(c1nc(C)oc1C)=O)OC N1(C(C2CC(=O)NC2)=O)CCC=C(C(=O)N2CCOC(C(=O)O)C2)C1 N1(C(c2cccc(CC)c2)=O)CCCCC(C(=O)NCC2CCN(C(C)C)C2)C1 CCC(C)C(=O)C(=O)N(CCCCC(=O)NCCn1ccccc1=O)C C(CCCC(CO)NC(C1CC2CCC(C1)O2)=O)NC(CC(C)F)=O c1(C(N(C)CC2(O)CCN(C(C(C)n3ccnc3)=O)C2)=O)cc2n(c1)CCSC2 N1(C(C(CCNC(c2cccc(C)c2N)=O)O)=O)CC2(C1)CC(C)(O)C2 C1(NC(c2c(CC)ocn2)=O)CC2CC1CN(C(c1c[nH]ccc1=O)=O)C2 c1(OCC(=O)NC(c2c(C)cccc2)C(C)(C)C)ccc(S(N)(=O)=O)cc1 C1(NC(C2CCCC23CC3)=O)CCN(c2nnc(C(F)F)s2)CC1F N1(C(C(CC2CN(C(c3cc(CC)sn3)=O)C2)F)=O)CC2CCOC(=O)C2C1 C1(C(=O)NC2C(Nc3cccc(C(=O)OCC)c3)CCC2)CC2(CCC2O)C1 CCC(C)C(C)C(=O)N1CCC(O)(CNC(c2ccc(C3CC3)s2)=O)CC1 CC(C)C(CC(=O)NN=c1cncc[nH]1)c1ccc(F)c(F)c1 N(CC(=O)COCCOCCOCCO)C(C=CC(C)=O)=O N1(C(c2ccc(C)cn2)=O)CC2(CNC(=O)CC(C)c3cccnc3)CC1CO2 C(=O)(C1CCCc2scnc21)N1CCC(NC(C(CC)C#N)=O)(CF)C1 C(=O)(N=c1c(Cl)c[nH]cc1I)C1C2(CCN(Cc3cnn(C)c3Cl)CC2)C1 c1(C(C)NC(C2COC2)=O)cccc([N+](=O)[O-])c1 CC(C)CC(C)CC(C)C(=O)NC1CC(C)(NC(c2cncc(CO)c2)=O)C1 C1(C)(CC(=O)NCC(c2ncc[nH]2)C)CCN(C(=O)CCN=[N+]=[N-])C1 C1(C(=O)NC(CC=C)CNC(=O)CC2CC(C3CC3)C2)CCCCC(=O)N1 C1(C)(C=O)CCCN1N1C(N(c2coc(Br)c2)C(CC(C)(C)C)=O)CC1 N1(C(C=C(C)c2cccs2)=O)CCCCCC1CNC(=O)CC12COC(C)(C1)C2 c1(OC)csc(C(=O)NCc2cn(C3CCN(C(=O)C(O)CF)C3)nn2)c1OC N1(C(CC(CC)C(F)F)=O)CCC2(CC1)CN(C(=O)CC1CNC(=O)C1)CCO2 c1(C(=O)NCCC2(O)CN(C(CC3(C=C)CCC3)=O)C2)sc2ccccc2c1C C(=O)(CN=c1cc[nH]cc1)NC(CCC)C(O)C(=O)Nc1cnccc1OC c1(C(=O)NC(CN(C(c2ccc(CC)s2)=O)CC)C)ccc2sc(O)nc2c1 C12(NC(CCC=CC)=O)CCC(CN(C(=O)C(F)(F)CCn3cccn3)C1)C2 c1(C(=O)NCC(C2CCC2)NC(CNC(C)=O)=O)cc2nc(Cl)ccc2s1 C(CCCNC(C1CC(N(C)C)C1)=O)N(C(C=C(COC)C)=O)C C(CN=c1[nH]c(=NCCCN(C)C(C)C)c2ccc(OC)cc2[nH]1)=CCCC c1(C(=O)NC(CC(C)C)(C)CNC(=O)CC2OCCCO2)cc2ccccc2s1 c1(C(=O)NC2C(C)C2C)c[nH]nc1CNC(=O)C=Cc1ccsc1 c1(C(=O)NC2CCCN(c3nc(CSC)c(Br)cn3)C2)cccc([N+](=O)[O-])c1I N1(C(c2ccn(CCCC)n2)=O)CCCC(C)(CNC(c2ccc(O)nn2)=O)C1 N1(C(C=C(C)Cl)=O)CC2CCCC1C2CNC(=O)CC1COC(=O)C1 Cc1ncc(C(N2CC(O)(CCNC(C34CC(C(F)F)(CO3)C4)=O)C2)=O)c(=N)[nH]1 C1(C(N)=O)(NC(C(C)Oc2ccn(C)n2)=O)CCC(C)(C)CC1 c1(NC(=O)CC2(NC(c3ccns3)=O)CCC2)cccc(-c2ccccc2)c1 C12(C(=O)OC)CCCCCC1N(C(c1nc(C(F)(F)F)cs1)C(=O)NC1CC1)CC2 Cc1cccc(C(=O)CC2(N3CC(n4cc(C5(C)CCCO5)nn4)C3)CC2)c1 CC1CCCC1(C(=O)NCc1cc(CO)on1)NC(=O)Cn1[nH]cnc1=N N1(C(C(CC(C)C)N(C)C)=O)CCc2sc(CNC(=O)CSC(F)F)nc2C1 C=CC1CN(C(=O)CC(=O)OCC)CC1NC(=O)CC(OCC)OCC C(=O)(C1=CC2(CCOC2)C1)NC1CCC(CNC(C(CSC)OC)=O)CC1 N1(C(C2C(C)CC=CC2)=O)CC(NC(=O)CNC(N)=O)CC2(CCC2)C1 c1(CNC(=O)Cc2ccco2)cnn2c1CN(C(c1cnc(C3CC3)s1)=O)CC2 N1(C(=O)NCC(CC)(C)c2ccncc2)CCn2c(C(C)(C)C)nnc2C1 C(C)(C(C(C)C)NC(=O)CC1CC(C)(C)C1)NC(c1cc(C)sc1)=O C(CCCCC(=O)NC1(CO)CN(C(C2CC(F)C2)=O)C1)N(C)C C1(C(N2CC3(CC(CNC(c4ccsn4)=O)OC3)C2)=O)CC2CC1C1C2C1(F)F c1(CC)nnc(C)cc1C(=O)NC1CC1CNC(c1cc(CC(C)C)on1)=O c1(CC)cc(C)c(C(=O)NC(C)(C)CCCNC(c2cc(=O)cc[nH]2)=O)o1 c1(C(=O)NC(C(C)C)CNC(c2ccc(F)nc2F)=O)ccc(F)c(Cl)c1F c1(C(N(C2CCN(C(C3CCC(=O)O3)=O)C2)CCC)=O)cccc(C(C)C)c1 C12(C(N3CCCC(N(C)C(c4nnn(C)n4)=O)CC3)=O)C3CCC(CC13)C2(F)F Cc1cc(C(N2CCC(F)C(NC(=O)CC3CS(=O)(=O)C3)C2)=O)cc(O)c1 n1(CC(=O)NCC2CC(C)N(c3cc(Cl)ncn3)C2)ccc(O)nc1=O c1(C(N2CCC(c3ccccc3)C2C(=O)O)C(=O)NC)ccc(Cl)cn1 C1(C(=O)NC(CC)(C)COC)CN(C(C2CCC2C#N)=O)CC12CCC2 Cc1cccn2c(=O)c(C(=O)NC3CCN(C(=O)CCC4CC4C)C3C)cnc12 C1(C(CNC(c2ccn(CC)n2)=O)(C)O)CCCN(C(=O)CP(C)(C)=O)C1 C1(C(=O)NC2(C#C)CCOC2)CCN(C(=O)C(C#N)(CC)CC)C(C)(C)C1 c1(CS(=O)(=O)NCc2cc(C(N3CCCC3)=O)on2)cccc(F)c1 C1(CNC(CCn2cnc(=N)[nH]2)=O)(CNC(=O)CN2CCCCC2)CCCCC1 c1(CNC(C2(C3N(C(C(CO)OC)=O)CCC3)CC2)=O)ncc(C)cn1 C=C(C)C(O)CC(=O)NCC(C)CNC(c1cccc(-n2cccn2)n1)=O N1(C(c2scc(CC)n2)=O)CCC2C(CCN2C(c2ccn(C(F)F)n2)=O)C1 c1(C(N2CC3(CCCN(C(C(C)(C)C#N)=O)C3)C2)=O)cc(=O)c2ccncc2o1 CC1CC(C(=O)NC2CCCCCC2C)CCN1C(C1CC(=O)CS1)=O N(C1C(=O)Nc2cc(Cl)ccc21)C(C1(C)N(C(CCc2cn(C)nc2)=O)CC1)=O c1(NC)cccc(C(N2CCOCC2CN(C(=O)CCCCNC(N)=O)C)=O)n1 c1(C(N2CCN(C(C(N3CCNC3=O)C)=O)CC2C)=O)nccc2ccncc12 C1(N(C(c2cn(CC3CCCCO3)nn2)=O)CC)CCC(NC(=O)C(N)=O)CC1 C1(CC(=O)NCCCCCN(C(C2(C(=O)NC)CCC2)=O)C)C(C)(C)C1(C)C c1(CCC=C)ccc(C(=O)NC2CC(O)(C(=O)NC3(c4cccs4)CC3)C2)cc1 C1(C(=O)NCc2cc(C(F)F)[nH]n2)(OC)CCN(C(=O)CC2CC2(C)C)C1 c1(NC(C2CCN(C(COCC(=O)OC(C)(C)C)=O)C2)=O)cc(F)cc(F)c1N N1(Cc2cnc(OCC)nc2)CCCC(C)(C(=O)N(C(C)C(F)(F)F)C)C1 Cc1cnc(C(=O)N(C(c2ccccc2)CNC(C2(C(F)(F)F)CC2)=O)C)cn1 N1(C(c2scc(OC)c2)=O)CCOC(CCCNC(C2(CO)CC2)=O)C1 n1(CC)cc(Cl)c(C(N2CC3(NC(C4OCCOC4C)=O)CC2C3)=O)n1 c1(C(=O)NCCN(C(c2c(C)occ2C(F)(F)F)=O)C)ccc(F)c(C(F)F)n1 CC(O)(CO)C(=O)NCCc1cn(-c2cccc(C(F)(F)F)c2)nn1 CN1CCC(C(=O)NCC2C(CNC(c3cc4sccc4[nH]3)=O)C2(F)F)CC1=O CCCC(C)(O)C(=O)N1CC(C(C)(C)O)(CNC(=O)CCC(C)CC)C1 CCCC(C)(C)C(=O)NC1CN(C(=O)C=CCN(CC)CC)CC1n1cccn1 CC1(C)CCCC(C(=O)NCCNC(=O)Cn2ncccc2=O)C1 N1(C(c2c(C)nc(-c3cc[nH]n3)s2)=O)C2CCCC1CN(C(=O)CCC1CC1)C2 C1(CNC(CCC(C)OC)=O)CC2(CCC2)CN1C(=O)CNC(c1cscn1)=O C1(C(=O)NCC2CCOC2=O)(NC(C(F)=CCC)=O)CC1(C)C C(CNCC1CCCO1)(C(C)(C)C)NC(C(n1ncc(C(=O)OC)c1)C)=O N1(C(CC2N(C(C)=O)CCC2)=O)CC(C)(C)CCC1CNC(=O)CN=S(C)(C)=O C(=O)(CCN=C(NCC(=O)N(C)OC)NCC(C)(C)Cc1cccc(Cl)c1)NC C(=O)(CCCCC(=O)NCCC(C)NC(=O)CCc1ccc2ocnc2c1)NC C(=O)(C(CC(=C)Cl)NC(=O)CCCCCc1ccccc1)NC1(C)CC(=C)C1 C(=O)(CCCCC(=O)N1CCN(C(=O)C(C)NC(=O)NC)CC1CCOC)NC N1(C(C2CC(C)NCC2)=O)CC2C=CC1CC2 CC(C)(C)CCC(=O)NCC1CCC(NC(=O)Cn2ccc(Br)n2)C1 c1(C(=O)NC(C2CCN(C(c3ccccc3)=O)C2)C)ccc(C(F)(F)F)nc1 c1(C(=O)NC(C2CCN(C(CC(=O)NC)=O)CC2)C)nc(=N)[nH]c2ccccc12 N1(C(C2(S(N)(=O)=O)CC2)=O)CCC(NC(=O)CC2CCCC23CC3)C2(CCC2)C1 CC(C)CC(C(=O)NC1CCC1NC(=O)C1=CCCOC1)N(C)C Cc1ccc2cccc(C(N3CC(CCNC(c4ncccc4N)=O)C3)=O)c2n1 C(=O)(C(C)(CNC(C1CCN(CC)C1)=O)CC)NCC(CCC)OCC S(=O)(=O)(c1c[nH]ccc1=NCC1CCC2(CC1)CC2)NCC(C(CC)C)O N1(C(C(C(C)C)F)=O)CCC(C)(C)C1C(=O)N(CC(C)(C)CN(C)C)C C1(CC=C)(CNC(=O)C(O)CN(C)C)CCN(C(=O)Cc2cnn(CC)c2)C1 S(=O)(=O)(c1c(Cl)cc(OC(F)(F)F)cc1Br)Nc1c(C(=O)OC)ccnc1SC C(=O)(C1=NOC(C(C)(C)C)C1)NC1C(C)CN(C(=O)CCn2ccc(=N)[nH]2)C1 n1(C(C(C)C)C)nc(-c2ccc(N(C)C)cn2)nc1C1COCCN1C C(=O)(C(C)CC(C)C)NCCC(=C)CNC(c1cnn(CC2CCCC2)c1)=O C(=O)(C1OCCc2ccccc21)N(CCNC(CSC(C)C)=O)C C(CS(=O)(=O)CC1CCC1)NC(c1c(Cl)n[nH]c1C)c1n(CCOC)nnn1 c1(CC(=O)NCC(C2CCCCC2)NC(=O)Cc2cc[nH]n2)sc(O)nc1O CC1(C)C(C(=O)NCC2COC(=O)N2)CCN1C(=O)C1CC1 N1(CCCc2ccc(NC(C(C)C)=O)cc2)CC(C)OCC1C C(C(F)(C(=O)NC1CCC(O)CC1)C(C)C)NC(CCNC(=O)OC)=O c1(C(=O)NCCN(C(CC(C)N(C)C)=O)CC(C)O)ccc2ccncc2n1 c1(CC(N2CC(F)CC(C(N3CCCC(OC)C3)=O)C2)=O)ccccc1[N+](=O)[O-] CC(CCN=C(NCC1CCC1)NC1CCC2(CC1)CC(CO)C2)N(C)C c1(C(=O)NCC(C(C)C)NC(C2CC2C(C)(C)C)=O)nccc2occc12 C1(C2CCCOC2)(NC(c2nnnn2C2COC2)c2ncoc2)CC1.C1CCC1 C1(C(=O)NCC(CC)N(C)C(c2nonc2N)=O)CCC(O)C1 Cc1ccc(C2CCCCC2NCCc2ccccc2C)c(C)c1 C(=O)(C(C)(C)CC(C)(C)C)NCC(C1CCN(C(C(C)C2CCC2)=O)CC1)(C)O c1(C(=O)NCC2N(C(c3n(CCC)ccc3)=O)CCC2)nc(OC)ccc1OC c1(CN2CCN(C(c3n(C)cnc3)=O)C3C2C3)cc(Cl)c(O)cc1F c1(CC2c3cn(nn3)CCN2)ccccc1Cl.C(=O)(CN(C)C)NC(=O)OC c1(C(N(CCN(C(C2(C#N)C(C)C2)=O)C)C)=O)cc(C2CCCC2)n(C)n1 N1(C(CNC(=O)OCC=C)=O)C2CCC1CC(OCCCOC(C)=O)C2 Cc1c(C=CC(=O)NC2CCC(N(C)C(c3cn(C)nn3)=O)C2)cnn1C S(=O)(=O)(c1ccc(Br)cc1NCCCn1ccnc1)N1C(C)(C)CC(O)CC1 N1(C(c2n(CCOC)ncn2)=O)CCC(c2cn(-c3ccc(F)cc3)nn2)C12CC2 c1(C(N(CCCNC(C=CCC)=O)CCO)=O)ccc2c(c1)CCCN2C(C)=O C12(NC(c3c(C)oc(Cl)n3)=O)CN(C(=O)C(O)c3ccsc3)CC1CS(=O)(=O)C2 N1(C(CN(C)CC)C)CCCC(C(=O)NCCN2C(C)CCC2C)CC1 CC1CCC(C(=O)NCc2cccc(F)n2)N1C(=O)CC1NC(=O)NC1=O C1(CC(=O)NCC(C)Cc2cn[nH]c2)CCCC1NC(c1ccncc1)=O N1(C(c2ccc(CSC)cc2)=O)CCC2CCCC12CNC(=O)CSC(F)F c1(C(=O)NC2CC3(C2)CC3C(=O)NC2CCCC2CN(C)C)cccc(O)c1F N1(C(COC(C)(C)C)=O)CCCC(CC(=O)NC2CC(CC(F)(F)F)C2)CC1 c1(OC)ccc([N+](=O)[O-])c(NCc2c(F)cc(Cl)cc2Cl)c1 CN1CCC(NC(=O)C(=O)N(CCO)Cc2ccoc2)C1(C)C CC1CC(CNC(c2cc(O)ncc2F)=O)CCN1C(=O)CS(C)(=O)=O Cc1ncn(-c2ccc(N3CCCC(C4CCCCO4)C3)nn2)c(=O)c1C c1(CC(N2CCC(CNC(C(CC=C)CC)=O)C2)=O)ccc2c(c1)CCCC2 c1(CC(=O)NC(C2CCCC2)CNC(CS(CC)=O)=O)ccc(S(C)=O)cc1 c1(C(=O)NCCC2CC(NC(CN3CC(=O)NC3=O)=O)C2)cn2c(n1)CCCC2 N1(C(COCC=C)=O)CCC(F)C(NC(=O)CSc2ccccc2Cl)C1 N1(C(C2C(C(=O)O)CCC2)=O)CCc2nc[nH]c2C12CCC2 N1(C(C(CC)F)=O)CC(C)CN(C(c2ccc3c(c2)CCN3C)=O)CC1C CCC(CC(=O)NC1CC(C)(CNC(=O)C=C2SCC(=O)N2C)C1)CC(F)(F)F C(=O)(C(C)CNC(=O)NCCc1n[nH]c(C)n1)OC.c1(C)ccccc1 Cc1cc2c(cc1C)OC(C(=O)NCC(F)CNC(=O)CCCNC(N)=O)C2 n1(CCCNC(CN(C(=O)OC(C)(C)C)C2CC2)=O)ncc(C(N)=O)n1.OC c1(C(=O)NC2CC(C)(NC(=O)CCc3nncs3)C2)sc2cc(F)ccc2c1Cl c1(C(=O)NCC(C)(C2CC2)NC(C(C)n2cncn2)=O)cc(N(C)C)ccn1 C#CCCCC(C)C(=O)N(CC(CC)NC(=O)CC1(COCC)CCOCC1)C CC(C)(CN1CCOCC1)C(=O)N1CCCC1CNC(C1CC(=O)C1(C)C)=O c1(C(=O)NCC2N(C(C3(CC)CCCC3)=O)CCC2)ccc(C)c(Cl)c1 C(C(=O)NC(CO)C1CC1)(C(C)(C)C)NC(c1cncc(NC)c1)=O C=CC1(NC(c2ccc(F)cc2)c2ccccn2)CCCC1 CCCCC(O)CCC(=O)N1CC2CC1(c1cn(CC3CC3C(F)(F)F)nn1)C2 C1(N(C)C)CCCN(C(=O)C(CNC(C2CCC3(CC3)C2)=O)CC2CC2)CC1 Cc1nc(Cn2cc(COCC3CN(C(=O)COCCO)C3)nn2)c(=O)[nH]c1C c1(C(N(C2CC(NC(C3C(CC)CCO3)=O)C2)C)=O)cccc(F)c1 c1(C(=O)OCC)cccnc1NCC1CCN(C(C2CCC(=O)N2)=O)CC1 CCCC(C(=O)N1CC=CC(NC(c2cc3cccnn3n2)=O)C1)S(N)(=O)=O CC#CCCCC(=O)N1CCC(N(CCO)C(c2cn(C)cc2C)=O)CC1 N1(C(CNC(CCCCC)=O)=O)Cc2ccc(CNC(=O)C(OC)OC)cc2C1 Cc1c(O)nc2ccccc2c1C(=O)NCC1CCN1C(=O)C(C)(O)C1CCC1 c1(C(=O)NC2CC(NC(C3CC34CCCOC4)=O)C2)cc2ccncc2cc1F C1(NC(c2ccc(Cl)s2)=O)CCN(C(=O)C(c2ccc(F)cc2F)=O)C12CC2 C(CC(C(C)(C)C)NC(C1(F)CC1)=O)N(C)C(c1ncoc1-c1cnn(C)c1)=O Cc1cc(C(N2CC(O)(C(F)C(=O)N(C3CCC4CC34)C)C2)=O)cn1C Cn1nc(O)cc1C(N1CC(F)CC1CNC(=O)C(c1ccccc1)O)=O CC(C)C(C)(Cc1ccccc1)NC(=O)C(=O)NC1CC(C)(C)C1 c1(CC(=O)NCCCN(C(C(CCC)=CCC)=O)C(C)C)cccc(Cl)c1F N1(C(c2c(CCC)cccc2)=O)CC2(CC(NC(=O)CS(N)(=O)=O)CO2)C1 Cc1cc(NNC(=O)NCc2ccccc2C#N)ccc1F c1(CNC(C2CC(CNC(c3cnc(C)o3)=O)OC2)=O)nc(C#N)cs1 C1(SC)CCCC1NC(=O)C(=O)NCC1CC(N)C1 c1(C(=O)NCCC(C)NC(c2c(C)onc2)=O)cc2c(Cl)nccc2s1 CC(C)CC(C(=O)N1CCN(C(=O)COCc2ccnn2C)CC(O)C1)C(N)=O n1(C(C)(C)C)cnc(C(=O)NCC(F)CNC(=O)C=C2CCSCC2)c1 C(=O)(CC(C)(C)SC)NCC(CC)NC(=O)C(C)C1(O)CCC1 N1(C(c2cc(OCC)no2)=O)CCCC(CCNC(C2(C)CC(C)=NO2)=O)CC1 C1(C(N2CCC(OC)(CNC(c3cccs3)=O)C2)=O)CC(S(C)(=O)=O)C1 Cc1ccc2nonc2c1C(=O)OCC(c1ccccc1Br)F C(CNC(=O)CCOCC1CCC1)(CC(=O)NC1CCOCC1O)OC C1(CNC(c2cnc3sccn23)=O)CN(C(=O)CC2CCOC2)C2COCC2O1 C1(NC(c2c(CC)n[nH]c2)=O)CCCC(NC(c2sc(C)cc2OC)=O)CC1 C1(C)(C(N2CC(CC=C)(NC(=O)C=CC(C)(C)C)C2)=O)CCCNC1=O C(=O)(C(C)(C)NC(=O)CCNC(=O)CCC1CCCOC1)N(C)C1CC1 c1(OC)cc(C(N2CCC(C(C)(C)NC(c3cnc(C4CC4)o3)=O)C2)=O)sn1 C(=O)(CC(C)(C)C(=O)NCC1C2CCC(C2)N1C(c1c[nH]nc1F)=O)OCC Cc1oc(C)c(C(=O)NC2CC3CC(NC(c4cncs4)=O)C2C3)c1C C(C)(CCCCNC(c1nnccc1C)=O)NC(C(CC)=CC)=O c1(C(=O)NC2CC3(CN(C(CCC=C(C)C)=O)C3)C2)cnc2cccnc2c1 N1(C(c2ccc(NC)cn2)=O)CCCC(NC(=O)Cc2cc(F)ccc2Cl)C1C O=C1CC(C(=O)N2CCN(C(C3CCCOCC3)=O)CC2CF)=NN1 CCCCCC(CC)C(=O)NC1CCC(CC(=O)NC2CN(CC)CC2C)CC1 N#CC1(C(=O)NC2CCCCCC2NC(C2(C3CC3)CCC2)=O)CCSCC1 c1(CC#N)ccccc1CCC(=O)NC(c1cn(Cc2cnn(C)c2)nn1)(C)C CC1(CNC(c2cc(Cl)cnc2O)=O)CCCN(C(c2coc3c2CSC3)=O)C1 C1(C)(CC(=O)N(C2(C(N3CC(O)(C)C3)=O)CCCC2)C)CCOCC1.C1(N)CC1 C1(C(=O)NC(CNC(c2cc(C)c(C)[nH]2)=O)(C)C(C)C)Cc2cccc(F)c2O1 C1(CC)CN(C(=O)Cn2cnnc2O)CCC1NC(=O)CCc1ccccc1C c1(C(=O)NC2CN(C(c3ccc(O)nc3)=O)CC23CC3)cc2cnccc2[nH]1 Cc1cc(F)ccc1CNC1CC(C(=O)NCC=CC2CCCCC2)C1 C12(CNC(C(CC)OC)=O)CC(CCO1)N(C(=O)C(C)Cc1cccnc1)C2 C(=O)(C1CCNc2ccc(O)cc21)NC(c1cn2ccccc2n1)C c1(C(=O)NCCN(CCOC)C(C2CCNC2=O)=O)c[nH]c(Br)c1 c1(C(N2CCC(NC(C(F)=CC)=O)CC2)=O)cc(S(N)(=O)=O)c(Cl)o1 c1(-c2cn(CC(CCNC(=O)Cn3cccc3)F)nn2)ccc(F)cn1 N1(C(C(C(C)C)SC)=O)C2CCC1CC(N(C)C(c1ccc(F)cc1)=O)C2 c1(C(=O)OC)ncc2c(Cl)cccc2n1.C12=CNC=CC1=NCCS2 C1(NC(CC2CC(OC)C2)=O)C2CC3CC(C2)CC1(CNC(=O)C1=NOCC1)C3 N1(C(C=CC(=O)N(C)C)=O)CCCC(C(=O)NCC2CC3(CCC3)CO2)(CO)C1 Cn1c(C(N2CC(NC(C3Cc4cscc4C3)=O)C(O)C2)=O)ccc1C#N c1(CNC(c2c(C)n(C)nc2)=O)ccc2c(c1)CCN(C(c1cncs1)=O)C2 C1(CN(C)C(C2(c3ccco3)CC2)=O)CCC(CNC(C2CC3CCC23)=O)CC1 C1(C(=O)NCC2(O)CC(CNC(CCCC#C)=O)C2)Cc2n[nH]cc2C(=O)N1 C(=O)(C1CCCn2nccc21)N1CCCC2(CN(C(C3=CCCC3C)=O)C2)C1 N1(C(C2N(N=O)CCC2)=O)CC(CNC(=O)CC2=CCCCC2)OC2CCCC12 Cc1c(C(=O)NC2CC(CNC(c3cc([N+](=O)[O-])n[nH]3)=O)C2)ccc2cncn12 C1(NC(C(CC)n2cncn2)=O)CC2(C1)CN(C(=O)CC(C)C(F)F)C2 Cc1nc2cccc(C(=O)NCC3C=CCN3C(c3ccncc3N)=O)c2[nH]1 C(=O)(C1=NOC(C)C1)N1CC(CCCNC(Cc2c(CC)con2)=O)OCC1 c1(NC(C2OCCN(C(C=NOC)=O)C2)C)ccc2c(n1)CCCC2=O N1(C(C(CNC(c2cn(C)nc2C)=O)OC)=O)CCCC(F)(CO)C1 S(=O)(=O)(CC1CCCc2ccccc21)N1C(c2cn(C)nc2C(F)F)CCC1 C1(C(N2CC(CNC(c3cnco3)=O)OCCC2)=O)CC2CCC1C21CC1 C1(C(=O)NCC(CC)NC(=O)CNC(c2ccccc2Cl)=O)CCC(C)(C)O1 Cn1nc(CNC(C2C3CCCC23)=O)c2c1CCN(C(C1CC3CCC1O3)=O)C2 c1(NC)c(C(N2CCN(C)CC2CNC(c2ccsc2Cl)=O)=O)cccc1F N1(C(C)=O)CCOC(C(N2CC(O)(CN(C(C3CCC4(CC4)C3)=O)CC)C2)=O)C1.C1CC1 n1(CC)cc(C(N2CC(O)(CNc3cc(F)ncn3)C2)=O)c2ccccc12 N1(C(C2CCCC(NC(C3(C)C=CCCC3)=O)C2)=O)CC2(CCOC2=O)C1 c1(Nc2cnc(C(=O)NC(C3CC(C(=O)OC)C3)=O)nc2)ccc(C)nc1CO c1(N2CC=CC(NC(Cc3cccc(C)c3)=O)C2)nc(C)ncc1C c1(C(=O)NC2CCC(OCC(=O)N(C3CC(OC)C3)C)C2)ncccc1C CC(C(=O)OC(C)(C)C)C(=O)NCC1(CO)CN(C(=O)C(=O)NC(C)C)C1 c1(CC)cc(C(=O)NCC2CC2NC(=O)COCC=Cc2ccccc2)c(C)o1 C(CCC1CC1)(C(=O)NCC(=O)NCC)NC(CCOCC#C)=O Cc1cn2c(n1)CC(C(=O)NC1CCCCCC1NC(C1C(C)C1C)=O)C2 N1(C(CNc2ccc(C)cc2)=O)CCN(C(=O)Cc2csnn2)CCC1C c1(C(=O)NC(c2nc(C)oc2C)C)cc(Br)cc(F)c1F n1(CCCSC)nnnc1C(c1cscc1SC)NC(c1nnc(C)o1)C N1(C(c2cc(C(C)C)[nH]n2)=O)CC2CCCC(C1)N2C(=O)C(c1csc(=N)[nH]1)=O S(=O)(=O)(c1ccc([N+](=O)[O-])c(Cl)c1)NC1CN(C(c2c(COC)onc2)=O)CC1F C1(C(=O)NC(C)CN(C)C(c2sccc2Cl)=O)CCCC2(C1)CC2(F)F c1(C(=O)NC(CNC(CC(C)OC)=O)C(C)(C)C)oc2ccccc2c1Br CCCC(C)(O)CC(=O)N1CC(C2CN(C(=O)C(F)=CCCF)C2)C1 N1(C(CC=CC=C)=O)CCC(C(=O)Nc2csc(Cl)c2OC)C(O)C1 N1(C(C(C(C)=O)(C)C)=O)CCC2(CCN(Cc3c[nH]c4ccc(F)cc34)C2)C1 c1(CC)c(C(N2CCC(C(C)CN(C(=O)CC)CC)CC2)=O)ccn1C C(=O)(C1=CCC(NC(=O)Cc2cc(C)on2)C1)N1C(CC)CC1 C(c1ccccc1Cl)=CC(=O)NCCCN(C(C(C)CC1CCCO1)=O)C C(=O)(N=c1cc2ccccn2[nH]1)C1C(C)(C)CN(C(c2cnnn2C2CC2)=O)C1 C(C1CCC(C)CC1)=C(C)C(=O)N(C1CC(NC(=O)C(C)CC(N)=O)C1)C C1(C(c2nnnn2C2CCC2)NCCN2CCCCC2)(OCC)CCCC1 Cc1ccc(C(=O)NC2(C)CCN(C(c3sccc3CO)=O)CC2)cc1C#N c1(NC(=O)Nc2ccc(-c3nnn(C)n3)cc2)ccc(C=O)cn1 c1(C(=O)NC(C2CN(C(c3cc(C#N)on3)=O)CCO2)C)ccc(F)c(Cl)c1F CCC(CC)C(C)C(=O)NC(CCOC)C(=O)NCCCC(F)F CC(C)C(C(=O)N1CCC1CNC(=O)C(C)NC(C1CCCC1)=O)C(C)C C(=O)(C(C)(C)CC(F)F)NCCCC(C)NC(C(C)CSC(F)(F)F)=O c1(OC)cc(OC)cc(CCC(=O)NCC2CCN(C(=O)C(Cl)=CCl)CC2C)c1 CC1(NC(C2CCCC(F)(F)C2)=O)CCN(C(=O)C2=CCCCO2)CC1 c1(C(N2CCN(C(CS(=O)(=O)NC)=O)CC2C(C)C)=O)cnc2ccc(C)cn12 C1(NC(=O)Nc2cc(C(=O)OC(C)(C)C)on2)CCN(c2ccccc2)S1(=O)=O C1(CNC(C=CC)=O)CN(C(c2cc(OC)nc(Cl)c2)=O)C(C)(C)C1 C1(NC(C=C2CCC(C)C2)=O)CCSC12CN(C(=O)CCC1(C)N=N1)C2 C1(C(N2CCCC(C(C)C)C2)C(=O)NCC)CCCC(C)C1 N1(C(COC(C)(C)C)=O)C2CCC1CC(NC(c1cc3ncsc3[nH]1)=O)C2 c1(CC2CCN(C(C3(C#C)CC3)=O)C2)cccc(C)c1.N12CC(C1)C2=O Cc1c(C(C(C)C)NC(c2cccc3sccc23)=O)oc2ccccc12 N1(C(CCc2c(C)ncs2)=O)CCCC(F)(CNC(c2coc(C(C)C)n2)=O)C1 N1(CCNC(C(CSC)C)=O)CCC(NC(C2(c3ccc(F)cc3)CC2)=O)CC1 N1(C(CSCC#C)=O)CCC2(CO)CN(C(=O)Cc3ccns3)CC2C1 c1(C(N2CC3(C(NC(CN=S(C)(C)=O)=O)CCC3)C2)=O)cc2c(O)ccc(F)c2[nH]1 C1(NC(CC2(C)CC2)=O)CC12CCN(C(=O)COC(=O)CO)C2 C#CCC(C)(CC)C(=O)NCC1CN(C(C2(C(=O)NCC)CC2)=O)CC(C)(C)O1 CCC(F)(F)CCNC(C(CC)CC)c1nnnn1C1CCOC1 C1(C(=O)NCc2c(CCNC(CSCCC)=O)ocn2)C2CCC1CC2 c1(C(=O)NCC2N(C(CC=C(C)C)=O)CC(C)CC2)ccc2c(=N)[nH]cnc2c1 C(=O)(C(CCC1CC1)NC(=O)Cc1ccnc(O)c1)NC(c1cn(C)cn1)C N1(C(c2cnc(CO)cn2)=O)CC(CNC(C2(CO)CCCO2)=O)CC12CCC2 c1(C(=O)NCc2c(C)n[nH]c2)cc(Br)c(O)cc1O c1(C(N2CC(NC(c3cc(CO)[nH]n3)=O)(CO)C2)=O)csc2ccncc12 C1(C(=O)NC2C(OC)CN(C(=O)CNc3ccccn3)C2)Cc2nnc(C)n2C1 N1(C(CN2CCN(C)CC2)=O)CCOC2(CCN(C(=O)CC#N)C2)C1 c1(C(=O)NCCCCN(C(C(c2c(C)cccc2)C)=O)C)c(Cl)nn(C)c1C N1(C(c2n(C)ncc2)=O)CCCN(C(=O)C(F)(F)c2ncccn2)CC1CO C(CNC(=O)C=C1CCC1)(C(=O)NC1CN(CC(F)F)C1)N(C)C c1(C(=O)NC2CCC(CC(=O)N(C(C)C3CC3)CC)CC2)cnn2c1OCC2 c1(C(=O)NCCC(C)N(C(C2C(C)(C(C)C)C2)=O)C)cccn2cnnc12 CCCC(CCCO)C(=O)N1CC2(CCCC2NC(c2cnc(CC)s2)=O)C1 N1(C(COCCC)=O)CCC2(CCCC2NC(c2c[nH]c3ccc(C)cc23)=O)C1 c1(N(CC(C(C)C)OC)C)nc(=NCc2ccc3ncsc3c2)[nH]c2ccsc12 c1(CN(C(=O)C(N2CCCC2CN2CCCCCC2)=O)CC)ccc(Cl)c(Cl)c1 Cc1cc(CNC(c2ccc(F)cc2)CC(C)C)cc2ccccc12 N1(C(C=C(C)C(C)C)=O)CCN(C)CC1CNC(=O)C(c1cscn1)N(C)C C(C1(C)CCOCC1)=CC(=O)NC(C)CC(C)NC(=O)CN(S(C)(=O)=O)C Cc1cc(C(=O)NC2CCCCC2NC(c2cnnc(C)c2)=O)n(C(C)(C)C)n1 c1(C(=O)NC2C(CNC(c3cnc4[nH]nnc4c3)=O)C2)scc2c1OCCO2 N1(C(C(COC)(C)C)=O)CCC2(NC(c3cncc(-n4cccc4)c3)=O)CC2C1 c1(C(=O)NC2C(CNC(c3nc(NC(C)=O)sc3)=O)CC2)cccnc1S N1(C(C(CC)OC)=O)CCN(C(=O)Cc2ccno2)C(CS(C)(=O)=O)C1 c1(OC)ccnc(O)c1C(=O)NC1CC(F)(CNC(c2ccc(CF)cc2)=O)C1 c1(C(CNC(c2cc(O)cs2)=O)NC(C2C(C)(C(C)C)C2)=O)ccccc1 c1(C(=O)NCCC2CC(C(N3CC(C(=O)N)C3)=O)C2)ccc(Cl)s1.CN(C)C C1(NC(c2cncc(C)n2)=O)CN(C(=O)CCc2cccnc2Cl)C(C)(C)C1 N1(C(CC=CCCCCC)=O)CCCCC1C1CCCN1C(c1ccc(Cl)o1)=O N1(C(C2N(S(CC)(=O)=O)CCC2)=O)CCCC(C)(NC(C2CC(O)C2)=O)C1 c1(CS(Cc2c(C)nc(CCN=[N+]=[N-])o2)=O)ccc2ccccc2c1 c1(CNC(C2CCC2F)=O)nccn1CC(F)F Cc1cccc(O)c1C(=O)NCC(F)CNC(c1ccsc1C)=O Cc1oncc1C(=O)NCC1CC(NC(=O)CCOCC(C)C)C1 CN1CCN(C(c2cn(C3CCC3OC(C3(CSC)CC3)=O)nn2)=O)C(CO)C1 CCCC(C)CCCC(=O)NCC1(CN(C(=O)CCN(C)CCO)C)CC1 CCC(C)C(C(=O)NCCCNC(=O)Cc1cn(C)nc1C)OC C1(CNC(c2ccn(CC)n2)=O)CCCN(C(=O)CSc2ccc(Cl)cc2)CC1 N1(C(c2c(OC)cccn2)=O)CCN(C(c2ccc(O)cc2)=O)CCC1C C#Cc1cc(C(=O)N(C2CN(C(c3cnnn3C)=O)CC2F)C)cc(F)c1 S(=O)(=O)(CCC(=O)N1CC(O)CC1CNC(C1CCC(C(=O)OC)C1)=O)N(C)C S(=O)(=O)(c1cccc(S(=O)(=O)N2CCC(c3cccnc3)C2)c1)N(C)C c1(NC(C)=O)cc(NC(=O)C(N2CCCCC2C(C)C)=O)ccc1Cl C1(CCNC(CSCC=C)=O)CN(C(=O)COC2CC2)CCS1(=O)=O N1(C(CC(C)N2CCCC2=O)=O)CC=C(CNC(=O)CC2(C)CC2(Cl)Cl)CC1 C1(NC(C=CCN(C)CC)=O)CC(OC)C12CCN(C(=O)C=C1CCCC1)CC2 c1(C(N(CCCNC(c2c(C)nccn2)=O)C)=O)ccc2c(n1)CCCN2 CC1=C(C(=O)NCC2CN(C(c3cccc(CO)n3)=O)CC2C)CCC1 Cc1cc(C(N2CCCC2(C)CNC(c2cc(C(F)F)ncn2)=O)=O)cnc1O c1(OC)ncnc(C)c1C(=O)NC1CC1NC(C1CC(=O)N(C)C1)=O C#CCC(C)(C(=O)NC1(CC(N)=O)CC1)NC(=O)C(C(C)C)SCC N1(C(C(=O)Cc2ccccc2)=O)CCC2(CCC2C(=O)Nc2ccccc2)CC1 c1(CNC(=O)NCC(=O)NCC(C2CC2)NC(C2COC(=O)C2)=O)ccccc1 Cc1cc(C)c(C(=O)NC2C=CC(C(=O)Nc3cc(F)cc(C#N)c3)C2)cc1Br Cc1ccc(C(=O)NCCC(C)N(C(=O)C(O)c2ccsc2)C)c(C(C)C)n1 C#CCC(CC#C)C(=O)NCC1CN(C(c2cccc(C(F)F)c2F)=O)CC1C C(=O)(C(C)(C)CC(F)F)NCC1(NC(c2cnc(CC)nc2C)=O)CC1 C1(NC(CN(C(=O)CSCC(N)=O)CCOC)=O)CC(CO)C1 N1(CC2C(C=C)C2)CCC(C(=O)NOC)CC1 C1(n2cc(CNC(=O)OC)nn2)CCCN(C(=O)Cc2cnn(C3CC3)c2)CC1 C(=O)(C(F)C(C)CNC(c1ncoc1CC)=O)N1CC(OCC#C)C1 C(=O)(C(F)C(C)(C)O)NC(CCCCNC(C(c1ccc(C)o1)C)=O)C N1(C(CCCCOCC)=O)CC2(CNC(=O)C(N3CCCC(C)C3)=O)CC1CO2 N1(C(c2ccc(NC(C)=O)cc2)=O)CC(NC(=O)C(O)CC(N)=O)C(C2CC2)C1 CC(CC(=O)NC1CC2CC(NC(=O)C(C)(C)N3CCOCC3)C2C1)C(F)F O=C(C1=CCCN(C(c2ccncc2)=O)C1)NCc1cc(C(F)(F)F)cc(F)c1 c1(C(=O)NCC2CCN(C(C(CC)(C)O)=O)C2)ccc2c(N)nccc2c1 C(=O)(C1=C(Cl)CCC1)N1CC(CC=C)(NC(c2cccnn2)=O)C1 C1(CNC(=O)CNC(=O)C(=O)Nc2ccc(F)cc2)CCCC2CNCC12 c1(C(=O)NCCC2CN(C(=O)C=C3CCCC3)CC(C)O2)snc2ccccc12 N1(C(c2scc(C)c2)=O)CCCCC1CNC(=O)Cc1ccn(CC(F)(F)F)n1 N1(C(c2ncc(NC)nc2)=O)CC(NC(c2cc(C)on2)=O)CC(O)C1 C(CC)(CCC(=O)N=c1ccn(C2CCC2)[nH]1)NC(C(CC#C)CC(F)F)=O C(=O)(C(C)(C)Cc1cccc(Cl)c1)N(CC(CNC(C(C)SCC)=O)C)C C(CC(CC)C(=O)N1CC(O)CC1(C)C(=O)Nc1cc(CC)ccc1C)=CC N1(c2cc(Nc3c(C)nn(CCOC)c3C)nc(C)n2)CC(C)(C)OC(C)(C)C1 N1(C(C(=O)NC(CC=C)CNC(=O)CC2CC(=O)C2)C)CCCCC1=O C(=O)(C(F)CC(C)(C)NC(c1cnc(C2CC2)o1)=O)NC1C(C)CC1 c1(CC(=O)NC2(C)CN(C(C(CC)SC)=O)C2)cccc([N+](=O)[O-])c1 C1(CC=C)(NC(C=CC)=O)CC2CCC(C1)N2C(c1cc2n(c(=O)c1)CCS2)=O c1(CC)cccc2c(C(=O)NC3CCN(C(=O)COC(C)=O)C(C)C3)c[nH]c12 C(=O)(C(CC1CCCC1)NC(C1CCCC1OC)=O)NCC1CC(=C)C1 N1(C(C(=O)N(C)C)=O)CC(NC(c2cn3cccnc3n2)=O)C2(CCC2)C1 CCCCCCCNC(=O)C(Cc1cnc[nH]1)NC(c1cc(O)nn1C)=O N1(C(C(CC)OC)=O)CC(CNC(c2nn(C)cc2Cl)=O)OC2COCC12 O=C(CC(O)C1CCCC1)NCc1c[nH]nc1C(=O)NC1CC(=C2CC2)C1 C1(c2ccccc2)(CNC(C(C)OCC)=O)CCN(C(=O)C(C2CC2)SC)CC1 C1(CNC(C(COCC)(C)C)=O)CC2(CO1)CN(C(=O)CCCN(C)C(C)C)C2 C12(C(=O)NCCC3N(C(C(CC#C)C4CC4)=O)CCC3)CCC(CC1)C(C)O2 CC1C2C(CCN2C(C2(CO)CC2)=O)CN1C(C1CCC(C#N)CC1)=O C1(NC(C(C(CC)C)O)=O)COC2(C1)CN(C(c1csc3nnsc13)=O)C2 N1(C(CCC(C)NC(C=CC=CCC)=O)=O)CCC(C)C(CO)C1 c1(OCCNC(C(N2CC(C)(C)C2C2CCCCC2)=O)=O)ccc(C#N)cc1 Cc1cccc(C(=O)NC(C)CCCNC(c2nc[nH]c2C(F)(F)F)=O)c1Cl c1(CNC2CC(CC(=O)Nc3c(C(=O)OC)cc(C)s3)C2)ccnc2[nH]ccc12 c1(C(N2CCC(NC(C=CCC)=O)C(CO)CC2)=O)c(C)cccc1[N+](=O)[O-] C1(COC(c2c(C3(C)COC3)noc2)=O)CC2(CCOC2)CO1 N1(C(CC2(C)OCCO2)=O)CC(NC(=O)CCc2ccccc2Cl)C2CC12 c1(OC)ccnc(O)c1C(=O)NCCC(C(C)C)NC(c1cnn2c1OCC2)=O C1(C(=O)OC)C(=O)NCCN1C(c1ccc(-c2ccco2)s1)=O c1(NCCN(CC)CC)ccc(S(=O)(=O)NCc2ncn(C)n2)c(Cl)c1 CCCC(C)(O)CC(=O)N(C)CCN(C(c1cncc(C(F)(F)F)c1)=O)C(C)C c1(OCC(N2CCC(NC(C3(C#C)CC3)=O)C2C)=O)cc(Cl)ccc1Cl C1(CC)CN(C(=O)C(COC)OC)CC1C(=O)N(CC(O)C1CCC1)C N1(C(c2ccn(CCC)n2)=O)CC(CNC(c2n[nH]c3c2CCC3)=O)C2(CC2)C1 N1(C(c2nnn(C(C)(C)C)n2)=O)CC2(C1)CN(C(=O)C(C)(C)n1ccnn1)CCO2 c1(CN(C(C=CC(C)NC(c2ccc(C)s2)=O)=O)C)c(C)noc1C C(F)(C(=O)NOC1CCCCC1)NC(CC1CC(N2CC(C)(OC)C2)C1)=O C(CC(=O)Nc1csnc1OC)(C(F)F)NC(c1n(CC)ncc1)=O c1(C(=O)NCC2C(NC(C3C(C)(C)C3)=O)C2)ccnc2[nH]c(CC3CC3)nc12 C1(C(N2C(CCNC(=O)CSc3cn[nH]c3)CCC2)=O)CCC(C2CC2)CC1 c1(NC(=O)Cn2ncnn2)cccc2c(C3CC3)cccc12 N1(C(=O)OC(C)(C)C)CC(NC2CCCC2)C(CC(C)(C)C)C1 N1(C(CC2(OC)CC2)=O)CCC2(CC(NC(=O)CSCCN(C)C)C2)C1 Cc1ccnc(-c2nc(Cn3cccn3)nn2C2CCC(C)C2)n1 c1(C(N2CC3(CC(NC(Cc4cnc(C)[nH]4)=O)C3)C2)=O)cccc2nc(O)[nH]c12 c1(N(CC(C)C)C)ccc(C(=O)NCCCC(C)NC(=O)CC2CC23CC3)cn1 C1(NC(c2csnc2Br)=O)(CO)CN(C(=O)C(C2CCCCC2)O)C1 N1(CC(C)O)CCN(C(C2CCN2)=O)CC1 c1(C(N2CCCCC(NC(C3N(C)CC(F)C3)=O)C2)=O)cc(S(N)(=O)=O)cn1C N1(C(c2c(C)onc2O)=O)CC2CC(C)N(C(=O)C(C3CCCCC3)O)C2C1 N1(C(C2C(NC(CCC3CC(C)C3)=O)CCO2)=O)CC(=O)NC(=O)C1C c1(CNC(=O)Nc2ccc(OCC#C)cc2)cnc(O)c(OCCN(C)C)c1 c1(CCN(C(=O)C=CC(N2CCNCC2)=O)C)cccc(F)c1 C1(CCNC(C2N(C(C)C)CCC2)=O)CCN(C(=O)Cn2cnccc2=O)CC1 C1(C(N(CCN2CCN(C(C=C(C)C)=O)CC2)C)=O)CCC(=O)N2CCCC12 CCCC(C(C)CC)(c1nnnn1CCCC1CC1)NC(C)CC(C)OC N1(C(C(=O)c2ccco2)=O)CC(F)(C(N2CCC(C(=O)O)C2)=O)C1 C1(C(=O)NC2CC=C(C(C)C)CC2)Cc2cc(Br)ccc2O1 C1(C(=O)NCC2N(C(CC3(C)CCC3)=O)CC2)CCC2(CCCC2)C1 CC1CN(C(c2cc(C(N)=O)[nH]n2)=O)CCN1C(c1ccon1)=O CN1CCC(C)(CNC(C2CCN(C(C3(C)CCCNC3=O)=O)CC2)=O)CC1 C(=O)(C(C)CC(F)(F)F)N1CCC(CC(=O)N)C1.c1(C2(CC)COC2)cn(C)nn1 C(CCCC(=O)Nn1cnc2ccccc12)NC(=O)C1=CCCCO1 N1(C(c2c(C)cc(C)[nH]2)=O)CC2ON=C(CNC(=O)Cc3nocc3C)C2C1 C(=O)(C(COCC(C)(C)C1CC1)N(c1ccccc1)C)OCCCN(C(C)=O)C N1(N(C(C(=O)OC)C)C)CC2(CCC2)C1C1CCOCC1 c1(SCC)cccnc1C(=O)NC1CN(C(=O)C(C2CC2)SC)CC1O CCCCC(O)CC(=O)N1CCC(C(C)(C)NC(c2cccc(C(C)C)c2)=O)C1 N1(S(C(C)C)(=O)=O)CC2(CN(C(C3CC3C3CC3)=O)CCO2)C1 c1(C(=O)NC2C(C)CN(C(=O)CC#N)CC2)ccnc2cc[nH]c12 C12(C(N3CCN(C(C(C)CC(N)=O)=O)C(CF)C3)=O)CC3CC(C(=O)N1)C2C3 C1(NC(c2c(CC)onc2C)=O)CC2CCC1N(C(c1ccc(CO)nc1)=O)C2 C(=O)(C1=NOC(C)(C)C1)NCC1CC(C)(C)N(C(C2CCCCO2)=O)C1 c1(C2(C(=O)NCC3C(NC(c4cc(C)sc4)=O)COC3)CC2)ccc(F)cc1Cl C(CC(C)C(=O)NC(c1nocc1C(=O)NOCC1CCCO1)C)=CCC c1(OCC)ccc(C)cc1C(=O)NC1(COC)CN(C(C2CCC2(C)C)=O)C1 N1(C(C(C)=C2CCC2)=O)C2CCCC1CC(NC(c1ccc(F)c(O)c1)=O)C2 c1(C(=O)NC(CC)CNC(=O)C(O)CCC(C)C)cc2c(OC)cccc2[nH]1 C#CCCCCC(=O)NC1CCOCC1C(N1CCC(=C)CC1)=O C1(C(C)C)CCC(N=c2[nH]c(=NC3CCCCC3C(C)C)[nH]c3c2CSC3)CC1 C(=O)(CCCCCO)N1CCC(n2cc(C3(C)CCOCC3)nn2)C1 CC1CN(S(=O)(=O)c2ccc(Br)s2)CCCN1c1ncc(C2CC2)cn1 Cc1cccc(C(N2CC3CC(NC(c4ncn(C)c4C)=O)C2C3)=O)c1Cl C(C(CC(C)C)C(=O)N1CC2CC2(CNC(=O)CC#N)C1)OC c1(NCc2nc(C(C)C)sc2)ccc(S(=O)(=O)N2CCCCC2CCO)cn1 C1(NC(C2CN(C(C)C)C(=O)C2)=O)CN(C(C2C3CC4C(C3=O)C24)=O)CC12CC2 Cc1oc2cc(C(=O)NCC3CC(CNC(C4CS(=O)(=O)C4)=O)CO3)[nH]c2c1C [N-]=[N+]=NCCCCCC(=O)NC1C=CC(C(=O)NCCC(O)C(F)(F)F)C1 C1(CNC(C=C(CC)C)=O)CC2(CCC2)CN1C(c1cnc(C(F)F)nc1)=O C=C(F)C1(CC(=O)NCc2ccc(CNC(=O)C(O)CF)cc2)CCC1 c1(N(C)C(C2CC(O)C2n2cccn2)=O)ccc2[nH]ccc2c1 CCC(C)(CC)C(=O)NC1CCCCC1CNC(=O)C(C)COC C(C)(CN=c1[nH]cnc2cccc([N+](=O)[O-])c12)(C1CC1)NC(C1C(C)(C)CC1)=O N1(C(=O)Nc2c(C)nc(N(C)C)s2)CC(C)(CO)CC1(C)C C(=O)(C#CC1(C)COC1)NCCn1ccc(C(=O)NCC(C)CO)c1 N1(C(N(c2cccc(C(F)(F)F)c2)C)=O)CC(F)CCC(F)C1 c1(OC)cc(OC)c(C(N2CCC(CN(C)C(c3csnc3C)=O)C2)=O)cc1Br C1(NC(C(=O)N(C(c2ccccc2OCF)C)C)=O)CCNCC(C)(C)C1 C12(NC(c3conc3C(F)(F)F)=O)COC(C1)C(NC(C1CC13CCCC3)=O)C2 c1(OCC(=O)NCC2N(C(COCCCC(C)C)=O)CCC2C)ccc(F)c(F)c1 c1(C(N2CC(CC(C)NC(C=CCC)=O)C2)=O)cc(Cl)cc2c1OCC2 c1(C2(C(=O)NCC(C)(C)NC(C=NOC)=O)CC2(F)F)ccccc1Br c1(N2CCCC(CC=C)(NC(c3cc(CO)oc3C)=O)C2)cc(C#N)nc(C)n1 S(=O)(=O)(c1cccnc1Cl)N1CC2(CN(C(=O)C(Br)Cc3ccccc3)C2)C1 C(=O)(C1=C(C)CCOC1)NC(CC(=C)Cl)C(=O)Nc1cncnc1OC c1(SC(C(=O)NCC(N(C(CCOCC#C)=O)C)C2CC2)C)nncn1C C(=O)(C(CC(C)(C)C)OC)NC(c1ccnn1C)C(=O)N(C(C)C1CC1)CC c1(C(=O)NCCC(C)NC(Cc2cc(C)[nH]n2)=O)ccnc2c1nnn2C C=CCC(F)(F)C(=O)NC(C)CC(C)NC(=O)CNC(=O)OC(C)(C)C C(=O)(CCCn1cccc1)NCCN(C(c1ccsc1C)=O)CC c1(OC)ccc(C(N2CCOCC2CNC(C2(CC3CCC3)CC2)=O)=O)c(C)n1 CC(C)CC(F)(F)C(=O)NC(C)CC1CCN(C(=O)C(F)OC(F)(F)F)CC1 C(=O)(C(F)(F)C(O)C1CC1)NCCN(CCC)C(C1C2CCN1CC2)=O Cc1nccc(C(=O)NCC2CC(C)(C)CN2C(=O)C(C)Cc2cnc[nH]2)c1C Cc1cc(C(=O)NCC2(C)CCN(C(=O)Cc3nccs3)C2)nnc1O C1(c2nnnn2C(C)(C)C)(NC(c2cncs2)C)CC2CCOC12 C(=O)(CCS(C)(=O)=O)N1CC(C(N2C(C)CC(F)C2)=O)C(C)C1 N1(C(c2cc(C(C)C)no2)=O)CCC2(CCN(C(=O)C(C)Cc3cnc[nH]3)C2)C1 c1(C(=O)NCCC(C)N(C(c2ncn(C(C)C)n2)=O)C)cc(O)cc(Br)c1 C1(C(N(C(C)CNC(=O)Cc2ccc(C(F)(F)F)cc2)C)=O)CCCCN1N=O CCCCC(CC)CCC(=O)NC(c1ccc(C)cc1)CNC(=O)C(O)C(C)C c1(C(=O)NCCC2(NC(C3C(C)C3C)=O)CC2)c[nH]nc1-c1ccc(Cl)s1 Cc1[nH]nc(C(N2CCC(NC(=O)CN(C)C(c3cccs3)=O)C2C)=O)c1C CC1CN(C(=O)CN2CC(=O)N(C)C2=O)CCC1NC(c1cc(Cl)nnc1O)=O CC(N=c1nc2c(ncn2C)c(NC2CC(=O)N(C)C2)[nH]1)c1cnc[nH]1 c1(CCC)nnc(S)n1CC(=O)NC(C1CN(C(c2cnc(C3CC3)o2)=O)C1)C C(C(N=c1nc2scnc2c(NCc2cc3n(n2)CCCO3)[nH]1)C1CC1)OC C1(C(N(C)CCNC(c2ccn(Cc3ccccc3)n2)=O)=O)COC(C)(C)CO1 c1(CCC(N2CCC(C)(CNC(C3(CCO)CC3)=O)C2)=O)nc2ncccn2n1 C1(C(N2CCN(C(c3ccc([N+](=O)[O-])[nH]3)=O)CC2CO)=O)CCc2nccn2C1 CC(C)C1=NOC(C)(C(=O)N(CCCNC(=O)C(C)NC(c2cccs2)=O)C)C1 C1(C(=O)O)(NC(c2cn(C)nc2C2CCC2)=O)CCOC(C)(C)C1 N1(C(C)C)CCCC1CC(N1CC(N(C(=O)CCOCC2CC2)C)C1)=O N1(C(c2c(SCC)nccn2)=O)CCCC(CC)(NC(=O)CN(C2CCC2)C)C1 N1(C(C2C(CC)C2)=O)CC2(C)CN(C(c3ccc(N)c(C)c3)=O)CC2(C)C1 N1(C(CNC(=O)Nc2ccns2)=O)CCC(NC(c2cncs2)=O)C(F)C1 n1(CCCF)nnnc1C(C1(n2ccnn2)CC1)NCc1ccnnc1 N1(C(c2c(C)oc(CO)c2)=O)CCC(NC(=O)CC2CCCN2C)CC(C)(C)C1 Cn1nccc1C=CC(=O)NCC=CC(=O)NC12CCC(C1)C2 c1(OC)c(F)ccc(C(N2CCC23CN(C(c2cc[n+]([O-])cc2)=O)C3)=O)c1F C(=O)(CC(C(F)F)NC(=O)CC=C)N1CC(CC#C)OCC1 c1(OCC)nc(C(N2CCC2CNC(C2CCCN2CC(C)C)=O)=O)co1 Cc1ccccc1-c1nc(CC2COCC2O)n(Cc2ccccc2F)n1 c1(CN2CCN(C3CCCN(C(CSC)=O)C3)C(=O)C2)ccc(C)cc1[N+](=O)[O-] c1(C(N2CC(CNC(C(CSC)C)=O)OC(C)(C)C2)=O)ccc([N+](=O)[O-])c(O)c1 N1(C(C(C)OCC)=O)CCC2CCC(NC(c3c(F)cc(F)c(F)c3F)=O)C1C2 CCC(C)(CNC(C1CCOCC1)=O)C(=O)NCC1(CCO)CN(C)C1 N1(CCC(=O)NC2C(NC(C3N(C)CCC3)=O)C2)C(=O)NC2(CCCC2)C1=O N1(C(C(C)C)=O)CCCC(C)C1CNC(C1(C2CCC2)CC1)=O c1(C(=O)NC(C(=O)NCCCCC#CC)CCC)ccccc1C#N c1(C(=O)NC2C(C)CN(C(=O)CCCn3ccccc3=O)C2)ccc(N)c(O)c1 C(=O)(CC(C)CNC(C1CCOCC1)=O)NC(c1ccncc1)CC Cn1cc(Br)c2c(N3CCC4(CCCCC4)CC3)ncnc12 N1(Cc2cnc(C(C)C)s2)CCC2(CC(C(=O)N3CC4OCCOC4C3)=NO2)C1 CC(C)(O)CC(=O)NC(CNC(c1cccc(OCCF)c1)=O)C1CCC1 c1(NC(c2cncc(NC(c3nc(CC)oc3)=O)c2)=O)cccc(Br)c1I N1(C(C2(COCC)CC2)=O)C2CCC1C(F)C(NC(c1nccnc1CC)=O)C2 C1(CC(=O)N(CCNC(=O)CSCc2n[nH]c(=N)s2)CC)CCN(C)CC1 C=CC(C)(C)CC(=O)NC1CCN(C(=O)Cc2cc(C)ccc2OC)C12CC2 c1(C(=O)NCC2CCN(C(CSCCCC)=O)C2)ccc(C)nc1OC C(=O)(C1CCCc2n[nH]cc21)NC1(CC=C)CCN(C(=O)C(C)(C)C(=C)C)C1 C1(NC(c2c(OC)nsc2)=O)CC2CC(NC(=O)COCc3cc(C)on3)CC12 C(CC(C(C)(C)C)NC(=O)CCCF)N(C)C(c1cnc(O)n1C)=O C#CC1CCCC(C(=O)NC2CSCN2C(=O)CC2CC3CC3C2)C1 CC1CCC(C)N1CC(N1CC(NC(C2CC23CCOC3)=O)C(C)C1)=O N1(C(C2C=C(C)CS2)=O)CCN(C(c2ccccc2CC#N)=O)C(C)C1 c1(C(=O)NC(C(CO)NC(Cn2c(C)nnn2)=O)C)ccc(CC2CC2)cc1 C1(C(=O)NCC(=O)N(C)C2CC2)CCC(C2CC2)N1C(=O)Cc1cscn1 N1(C(c2c(OC)nc(C)cc2)=O)CCC2(CC(NC(c3cc(Cl)no3)=O)CO2)C1 N1(C(C=C(C)c2ccsc2)=O)CC(CNC(=O)C=Cc2nc(C)cs2)CCC1C n1(CC(=O)NCC(C)N(C(=O)CCc2cnn[nH]2)C)cc(C2CC2)nn1 C(=O)(CC(C(C)OC)NC(=O)Cc1ccnn1C)N(CC)Cc1ncc[nH]1 N1(C(c2ncn(CC)n2)=O)CCOC(C(C)NC(=O)CC2(O)CCC2)C1 CC(CN(C(=O)CCc1ccccc1)C)N=c1cc(C2CC2)nc(S(C)(=O)=O)[nH]1 C1(CNC(c2cn(CC)nn2)=O)CN(C(c2ccc(CO)nc2C)=O)CC1(F)F C1(NC(C)=O)CN(C(c2cn(CC)nc2)C(=O)Nc2ccccc2)CC1O c1(OCC#C)ccc(C(=O)NC2CC2NC(=O)C(F)(F)c2csc(C)c2)cc1 Cn1cc(CN2CCC(c3ncc(C(=O)O)s3)CC2)c(O)nc1=O c1(OC)ccnc(C(=O)NC(C)(CNC(c2ccc(C)cc2F)=O)C(C)C)c1C Cc1nc(NCC(C)C2CCC2)cc(=NCc2cccc(F)c2F)[nH]1 c1(C(=O)NC(C(C)NC(c2cc(=O)cc[nH]2)=O)C)cc(C(F)(F)F)ccc1F C=C1CCN(C(=O)CC2CCC(C(=O)NC)CC2)C(C(=O)NOCCO)C1 c1(C(=O)NCC(CC(=O)NC(C#C)C)OC)ccc2[nH]ccc2c1 Cc1cc2nc(C(=O)NC(C)CCNC(=O)CCn3ccnn3)cn2cc1C C1(F)(C(N2CCC(OCC(N)=O)C2)=O)CCCN(C(C2CCSCC2)=O)C1 C(=O)(CC(C(C)OC)NC(=O)C(C)(COC)N(C)C)NCC(CCC)OC c1(Nc2c(C(=O)Nc3cccnc3CO)scc2)ncnc2c(Br)cccc12 CC1(CNC(C2CCCCC2O)=O)CCCN1C(=O)C=Cc1cccnc1 c1(C2C(C)O2)csc2ccccc12.CC(CS(=O)(=O)N(C)C)Oc1cccc(F)c1 c1(C(=O)NCC2C(NC(c3ccc(C)n3C)=O)CCCC2)ccc(Cl)c(F)c1N N1(C(CCSc2n(C)nnn2)=O)CC2(COC(CNC(=O)CNS(N)(=O)=O)C2)C1 N1(C(CC2(COC)CCCC2)=O)CCC(OC2CN(C(=O)CNC(C)=O)C2)CC1 c1(SCC=C)ccccc1C(=O)NCCCC(C)NC(C1CCC(=O)O1)=O C12(C(=O)NCC34CC(CC)(N(C(=O)C(C)=CC5CC5)C3)C4)CCCCC1OCC2 C1(C(N2CCCC(C(NOCCC)=O)C2)=O)Cc2nccn2C1 CC1CN(C(c2ccc(Oc3ccccc3)o2)=O)CC1NC(=O)C(C)N(C)C Cc1nn(C)c2ccc(C(=O)OCC3CCc4nccn4CC3)cc12 N1(C(CC(C=C)(C)C)=O)Cc2ccccc2C1CNC(=O)CSS(C)(=O)=O C(=O)(C1Cc2ccccc21)NCCOCCOCC(N1CCC(C)(O)C1)=O N1(C(CC2C(NC(C(C(=C)C)(C)C)=O)C2)=O)CC(O)C(N=[N+]=[N-])C1 c1(C(N(C(C)CNC(C2(F)CCOC2)=O)CC)=O)cn(C2CCCC2)nn1 N1(C(c2cnc(OC)nc2C)=O)C2CCC1C(F)C(NC(C1CC(C)(C)C1)=O)C2 c1(CC)c(C(=O)NC2CC(CNC(=O)C(Br)=C(C)C)C2(C)C)[nH]c(C)c1C(N)=O CC1(C(N2CCCC2C2CCOC2)=O)CCN(C(c2csc(Cl)n2)=O)CC1 N1(C(CCCCSC)=O)CCN(C(=O)Cc2cc(C)ccc2C)CC1C C1(C)(N(C)C)CCN(C(=O)COCCNC(c2ccsc2Cl)=O)C1 C(C(CCO)NC(C1CCCN1C(c1cscn1)=O)=O)OC N1(c2ncc(C)c(C)n2)CCCC2(NC(c3ccn(C)c(=O)c3)=O)CCCC12 CCC(CC(=O)N1CC(OCCC(=O)NC2CC(C(C)O)C2)C1)CC(C)C C1(C(=O)NCC(C)(C)CNC(=O)Cc2ccc(O)c(Cl)c2)CCC2(CCC2)OC1 C1(C(=O)NC(CC(=O)NC)C)CC2CC2N1C(c1ccccc1NC)=O C(=O)(CCC(=O)C(C)(C)C)NC(CCOC)C(=O)NCCC1CCCC(C)C1 C1(CC)C(C(=O)N(CCO)CCO)CCN1C(C1SCCS1)=O CC(CC(N)=O)C(=O)NCCC1CCN(C(c2cc(-c3ccco3)on2)=O)C1 c1(OC)cc(NS(C)(=O)=O)ccc1NC(=O)Nc1nnc(SC(F)(F)F)s1 C(CCC(O)C(=O)NCCN1CC=CCC1)NC(C(C)CCN(C)C)=O CN1CCN(C(c2cc(O)nc(O)n2)=O)C(CNC(C23CCCN2CCC3)=O)C1 N1(C(C(C)CNC(N)=O)=O)CCCC2(CNC(=O)CN3CC4CC4C3)CCCC12 C1(NC(CCOCC#C)=O)(CNC(=O)CNC(=O)C(C)CC)CCCCC1.C(C)(=O)O c1(C(=O)NC(CN(C(C2CCC(=O)N2C)=O)CC)C)cc(Cl)cc(Cl)c1N c1(C(N2C(C(=O)Nc3c(C)c(Br)ncc3)CC(F)C2)=O)ccc2n[nH]cc2c1 C1(CNC(C(CC)OC2CCCCC2)=O)CCCN(C(C2CC=CCO2)=O)CC1 Cc1nn(C2CCC2)cc1C(=O)NC1CCC(N(C)C(c2cc[nH]c2)=O)CC1 c1(C(N2C(CNC(Cn3c(C)nnn3)=O)CC2)=O)snc(-c2ccccc2)c1N C1(OC)C(O)CC1N=c1nc(N2CCC=C(F)C2)c2c([nH]1)CCCCCC2 CS(=O)(=O)C1(C(=O)NC2CN(C(=O)CSC3CCOC3=O)CC2O)CC(O)C1 C(=O)(C(O)CCCNC(c1nnn(CC)c1C)=O)NC(c1noc(C)n1)CC c1(OCC(=O)NCC2(NC(C3CC=CCO3)=O)CCOC2)c(Cl)cccc1Cl C(CC(O)CC(=O)NCC(C(C)C)NC(c1cc(C(F)(F)F)ccc1N)=O)SC N1(C(CN(C(C)=O)C)=O)CCC2(CCCN2c2ccc3nnnn3n2)C1 N1(C(CCSCC)=O)CCN(C(C2CCCC23CCC3)=O)C(c2ccccc2)C1 C=CCCCCCCNC(=O)C(CC(C)C)ONC(=O)CCOC(C)=O CC1(C2CC2)CN(C(=O)CC2CCC(NC(=O)CN3CCCC3=O)C2)CCO1 CCCC(CCC)=CC(=O)NC1CC(C(=O)N(C(C)C(=O)OCC)C)CC1O C(C(CNC(C1(C2(C)CC2)CC1)=O)S(C)(=O)=O)NC(c1n(C=C)nnc1)=O N1(C(C(CC=C)C)=O)CCC2CN(C(=O)C(C)(C)F)CCC12 C(=O)(C1=C(C)OCC1)NC1C(OC)CN(C(c2c(C(F)(F)F)cc[nH]c2=N)=O)C1 N1(C(c2ccc(CCCC)o2)C(=O)NCc2cccs2)CCC(OCC)C(C)C1 C1(C(=O)NC2CCN(C(CC3(C=C)CC3)=O)C2)Cc2ccccc2S1(=O)=O S(=O)(=O)(CCCCS(=O)(=O)N1CC(C#N)C1)N(C)Cc1c(C)nccn1 C(c1cncnc1O)=CC(=O)N(CCC(C)NC(c1cncc(OC)n1)=O)C C(=O)(C1=Cc2ccccc2C1)N1CC(C)C(NC(C(F)=C(C)C)=O)C(C)C1 c1(CNCCCc2c(C)ccnc2)cn(C)c2ccc(Br)cc12 N1(C(C(C)NC(N)=O)=O)CCCN(C(=O)C(F)Cc2cccs2)C(CO)C1 C1(NC(C(C(CC)C)OC)=O)CN(C(=O)C=Cc2cncnc2O)CC1C1CC1 N1(C(CN(CCOC)C(C2CCCCC2C)=O)=O)CCC(C)(CO)CC1 c1(N2CC(C(C)NC(C3CCCCN3C3CCCC3)=O)C2)cc(O)nc(=O)n1C c1(CNC(C(=O)N(C(CSC)C)C)=O)c(F)c(F)cc(F)c1F C1(C(=O)NCC2(F)CCN(C(c3n(C(C)C)ccn3)=O)C2)CC(C2CCC2)C1 c1(C(=O)NC(CC2CN(CC(C)=CC3CC3)C2)C)ccc(S(C)=O)cc1 CCCCC(C(=O)NCC(F)CNC(c1ccccc1SC(F)F)=O)NC(N)=O CC1(C)CC(CC(=O)NC2CCOC2)CN1C(=O)CCC(F)(F)F C(CCC)(C(O)C(=O)N1CCS(=O)C(C)C1)NC(C(CC=CC)CC)=O N1(Cc2c(C)ccc(Br)c2)CCC2CC(C(=O)NC3CCC(C#N)CC3)C2C1 c1(C2(C(N(C(CNC(c3cnn(C)c3)=O)C3CC3)C)=O)CC2)ccc(F)nc1 C1(NC(=O)Nc2cccc(-c3nc(C)on3)c2)CC(C)N(C)NC1=O C#Cc1cncc(C(N2CCC(C(CO)NC(=O)C(C(C)CC)OC)CC2)=O)c1 N1(C(C(C)OCCOC)=O)CC2(CC(NC(c3nc(Cl)sc3Cl)=O)CO2)C1 N1(C(C(C)CC(C)(C)C)=O)CCC2CCN(C(c3ccc(CCF)cc3)=O)C2C1 c1(C(C2C(C)=CCCC2C)NC=C(F)F)cc([N+](=O)[O-])ccc1Cl O=C(C(O)C(CCO)c1ccccc1)Nc1ccccc1C1CCC1 CCC1=C(C(=O)NCC2(NC(=O)C(C)CSC(F)(F)F)CC2)CCCO1 C1(C)(NC(C(c2cccc(Br)c2)OC)=O)CCN(C(=O)CCCN(C)C)C1 N1(C(c2cc(CCC)nc(O)c2)=O)CCC2(CCCN2C(c2ncoc2C)=O)C1 c1(C(=O)NC2C(CNC(c3ccc(CC)o3)=O)C2)ccc(C(F)F)cc1OC c1(C(=O)NCC2(O)CCCN(C(C3(C)ON=C(C)C3)=O)C2)nccc2[nH]ccc12 N1(C(CC2CC(NC(C(COC)OC)=O)C2(C)C)=O)CC2CC(C)(C)C2C1 C1(Cc2c(Cl)cccc2Cl)CN(CCNC(c2c(C)nccc2)=O)CCC1F Cn1c(C(=O)NC2(C)CC2)ccc1C1COCCN1C(c1ccns1)=O CCCCC(C(=O)N(CCCC(C)(F)F)C)NC(c1ccnc(OC)n1)=O C#CCCC(C(=O)OC)NC(=O)C(C)N(C(=O)CC1CC(=C)C1)CCC c1(CC)nc(C(=O)NC2CCN(C(c3ccccc3O)=O)C2)c(C)o1 c1(C(N2CC(C)C(NC(=O)CCCc3csc(=N)[nH]3)C2)=O)ccn2nncc2c1 C1(C(=O)NC2CC(CN3CCCCC3)C2)(NC(CC(=O)OCC)=O)CCOCC1 C1(NC(CCCSC)=O)CN(C(c2cc(F)n[nH]2)=O)CCC1C CS(=O)(=O)c1ccc(C(=O)Nc2ncc(I)cn2)cc1Br N1(C(C2C(C)(C)CCCC2)=O)CCC2(CC1)CC2C(N1CC(C(F)(F)F)C1)=O c1(NC(=O)NC(c2ncc(C)[nH]2)C(C)(C)C)cnn(CCO)c1C c1(C(=O)NCC23CCCN(C(COC)=O)C2CCC3)cc(Cl)c(Cl)c([N+](=O)[O-])c1 c1(OC)cc(C(=O)NCCCCNC(C2C3CCC(C3)C2(C)C)=O)cc(Cl)c1O C#CCCCCC(=O)NCC1(Nn2cc(C3(C)CC(F)(F)C3)nn2)CC1 c1(C(C)=O)cccc(C(N2CCC(F)(CNC(C3(C)CC(C)=NO3)=O)C2)=O)c1 C1(NC(c2c(C)csc2Cl)=O)CC2CC(NC(C3CCOC3)=O)C2C1 C(=O)(CC(C)(C)C(=O)NC1CN(C(=O)C(C)C2=CCCC2)CC1C(F)(F)F)OC c1(NC(C2(CC)CC(C(=O)NC(C)C(C(C)C)SC)C2)=O)cc2ccc(Cl)cc2s1 CC(C)CC(C)CC(=O)N1C2CCC1CN(C(C1CCc3ncnn3C1)=O)C2 N1(C(CCCC#N)=O)CC2(CCC2)CC1CNC(C1CCCCN1CC(F)F)=O CC1(C)C(=O)CC1C(N1CCC(CNC(=O)CSCCc2ccccc2)C1)=O Cc1ccc2oc(C(=O)NC3CCC3NC(c3ccc(CN(C)C)o3)=O)cc2n1 N1(C(C2(NC(C(CC(C)C)O)=O)CC(CO)C2)=O)CCOCC(C)(F)C1 N1(C(C(C)(C)OC)=O)CCC2CCN(C(=O)C(C#N)C(C)(C)C)C2C1 c1(C(=O)NC2C(NC(C(C)Cc3ccc(C#N)cc3)=O)C2)ccnc2cc[nH]c12 N1(C(c2c(C)onc2C2CC2)=O)CCCCC(NC(C2C3CC4C(C3)C24)=O)C1 N1(C(C2CCCC(C)(C)C2)=O)CCC2CCN(C(=O)CCC(C)(C)[N+](=O)[O-])C2C1 c1(C(=O)NCC2C(NC(=O)COC3CC=CC3)CCCC2)cc(F)cc(Cl)c1 c1(C(=O)NCC(CCOC)NC(C(C)OCC=C)=O)cc2ccccc2nn1 C1(CNC(CCN(CC)CC)=O)CCC(NC(=O)CCn2cc(C)cn2)C1 CC1CCN(C(c2cnn(CC3CCCC3)c2)=O)CC1NC(c1nsnc1O)=O CC1(C)CCN(C(=O)C2=CCCSC2)CC1CNC(=O)COC1CCOC1 C1(C(=O)NC2(CN(C(=O)CCC3CC3(Cl)Cl)C)CC2)Cc2cc(F)cc(F)c2O1 CCC(CC(=O)NCC(CC1CC1)OC)NC(=O)C(C)N=[N+]=[N-] c1(C(=O)NCC(CNC(C2C(C)(C)CO2)=O)F)ccc2cc(O)ccc2c1 N1(C(c2nc(C)on2)C(=O)NCC2CC2)CC2C(NC(=O)C(F)(F)F)C2C1 C1(NC(CC(=C)C)=O)CCC2CN(C(=O)C(C)=C3CCCC3)CCC2C1 CCC(C(=O)NCC1C=CC(NC(c2cccnn2)=O)C1)Sc1ccccc1 Cc1ccc(F)cc1C(N1CCC(CC(=O)Nc2csc(C3CC3)n2)CC1)=O c1(C(N(C)Cc2cn(CCC(C)C)nn2)=O)nc2n(c1C(=O)O)CCCC2 N1(CC(=O)NCC)CCc2cc(F)c(F)cc21.c12ccc(Cl)cc1C(=O)N2C C1(NC(C2(NC(C(CC3CC3)OC)=O)CC(F)(F)C2)=O)CCCC(O)CC1 c1(C(N2C3CN(C(C(C)=CC4CC4)=O)C(C3)C2)=O)cc2c(cc1Br)CCN2 C1(OC)CN(C(=O)CCc2cnoc2)CC1C(=O)N(C1CCC(O)CC1)C Cc1cc(NC(C2CC2C)=O)cc(C)c1.Cc1nc(C(=O)N(CC)C2CC2)cs1 C(=O)(C1=CCCCCC1)NC(C)C(C)(C)C(=O)NC(Cc1cnc[nH]1)CO C1(CNC(c2cc(C)ncn2)=O)CC2(CCC2)CN1C(=O)C=Cc1ccc(Cl)s1 c1(C)ccccc1OC.C(C(C)C(=O)NCC1(NC(C2CCCCC2)=O)CC1)OC c1(C(N2CCC(OC)C(C)C2)C(=O)NCCOC)nc2ccc(Br)cc2s1 C1(C(=O)NCC2CN(C(=O)CCOc3cccc(Cl)c3)C2)CCS(=O)(=O)CC1 CC(C(=O)N1CCN(C2CCCN(C(=O)COCCN(C)C)C2)CC1)C(C)(F)F N1(C(C(C)OCC#C)=O)CCC(CO)C(NC(c2cnnn2C)=O)C1 N1(C(c2n(C)nc(C(C)(C)C)c2)=O)C2CCC1CN(C(c1cc(F)cs1)=O)C2 Cc1cc(CN=C(NCC(c2nccs2)C)NC2CCS(=O)(=O)C2)ccc1F c1(-c2n(CCCSC)c(N3CCC(C)(C)CC3)nn2)cc(Cl)c2c(c1)OCO2 CN1CCC(NC(c2cc(C(F)F)n(C)n2)=O)C12CCCN(C(C1(F)CC1)=O)C2 N1(C(=O)Nc2ccc(CC3CC3)cc2)Cc2nnsc2C1 c1(CNC(C(CCOC)OC)=O)nc2c(s1)CCN(C(c1c(C)cnn1C)=O)C2 c1(C(=O)NC(CCOC)CNC(C2CC(=O)N(OC)C2)=O)csc2ccccc12 C(=O)(CCC(=O)N(CCCCN(C(=O)CC1CC(CC)C1)C)C)OCC CCCCC(CC(=O)N1CCC(COC)CC1)NC(C1C2C3CCC(C3)C12)=O c1(C(=O)NC2CN(C(C(CC)C(F)(F)F)=O)CC2(C)C)ccc2c(ccn2C)c1 C1(C(N(C)CC2CC(F)(F)C2)=O)CCN(C(C2CCCC23CCC3)=O)CCO1 C(C(C)(C)C(=O)NCCCCN(C)C1CC1)N(C(C(COC(C)=O)C)=O)C C12(C(=O)NCC(F)CO)CC(CN1C(=O)C(C1CCOCC1)F)C2 Cc1oc(C#N)cc1C(N1CC(NC(C23CCC(CC2)CC3)=O)CC(C)C1)=O c1(C(C(N2CCC(CN3C(=O)C3)C2)=O)O)cccc(Cl)c1.Cn1ncnc1C C#CC(C)(C)C(=O)NC1CCN(C2CCN(C(=O)C(C=C)c3ccccc3)C2)CC1 C1(C#N)(C(N2CC(CNC(c3cc(SC)c(F)cc3)=O)C2)=O)C(C#N)C1(C)C C(=O)(C1CCCc2nc[nH]c21)N(CCCCNC(=O)CN1CCCCCC1)CCO Cc1c(NCCCN2CCOC2=O)ncnc1N(C)Cc1ccc(C2CC2C)o1 CC(C)(C)C1=NOC(C)(C(N2C3CCC2CN(C(=O)CNC=O)C3)=O)C1 N1(C(CNC(c2ccn(C)n2)CC)=O)CCC(N=[N+]=[N-])(C(=O)NC(C)C)C1 C(C)(C1CCCc2cccnc21)NC(C1(C)CN(C(=O)OC)C1)=O C(=O)(C(C#N)C(C)(C)C)NC1CCN(C(CCSC)=O)C1C Cc1ccc(C(C(=O)NCC(C)C)N(C2CCC2C)C)cc1I c1(C(=O)NCC(C)CN(C)C(C2CCN3CCOCC23)=O)ccn2ccnc2c1 N1(C(C2(C#N)CCC(=O)C2)=O)CCCC(O)(Cn2cc(CCCCO)nn2)CC1 C1(NC(C(CC)SC)=O)CCCC12CCN(C(c1ccc(NC)c(F)c1)=O)CC2 C1(NC(CN(CCOC)C)=O)CC2(C1)CC(C(=O)NCC(F)(F)C(C)C)C2 Cc1oc(C#N)cc1C(=O)NC1CC(NC(=O)C(C)OC2CCCCC2)C(O)C1 C1(CC(N2CCCC(C(CC)N(C)C)C2)=O)CC(C)N(C(C)=O)C1 c1(C(=O)NC(CC#C)(C)C(=O)NCC(Cl)C(C)(F)F)ccc(C#N)cc1C c1(-c2cc(OC)c(F)nc2)ccc2[nH]c(C(=O)Nc3ccc(F)nc3)cc2c1 c1(CC(N2CC(n3cc(CCN(CC)CC)nn3)C(C)C2)=O)ccc(F)cc1C Cc1ccc(C(=O)NCCOCCC(=O)Nc2cnc(O)cc2C)c(C)n1 C1(N(C)C(c2ocnc2C(F)F)=O)CN(C(c2cn(C)[nH]c2=N)=O)CC12CC2 C=CCC(CC)C(=O)N(CC(CC)NC(c1ccc(F)c(NC(C)=O)c1)=O)CC N1(C(C2ON=C(C)C2)=O)CCOC(C)C1C(=O)NOCCOCCO C(=O)(C1CCCc2sccc21)NCCNC(c1ccc(-c2nc(C)c(C)o2)cc1)=O N1(C(C2Cc3c(nc(C)[nH]3)CC2)=O)CCCC(N=c2[nH]c(Cl)nc(C)c2Cl)CC1 C1(NC(c2nc(C(C)OC)sc2)=O)CN(C2CCC2)CC1C.C12(CC1)C(=O)NC2 N1(C(C(C)OCC=C)=O)CC(OC)CC1CNC(=O)CC1(CO)CC1 C(=O)(C(F)(F)C(O)C1CC1)N(CC(CC)NC(=O)CC1(C)CC1)CC N1(c2c(F)cc(N3CCOCC3)cc2F)CCc2cc(Br)c(F)cc21 C1(NC(C(C)NC(C2CCC2)=O)=O)CN(C(=O)C2=COCC2)CC2(CC2)C1 Cc1c(Cl)c(C(=O)NCC2CC2NC(=O)C(C)N(C)C)nn1C c1(C(=O)NC2CCN(C(c3c(C)cc(O)cc3)=O)C2C)cn(C)c(=O)n(C)c1=O S(=O)(=O)(c1ccc(NC2CCCSCC2)nc1)N1CCS(=O)(=O)CC1 c1(C(N(CCC)CCNC(=O)C(n2cc(Br)cn2)C)=O)cccc(CO)c1C C=CC(C)CC(=O)NCC(C)(C)CCNC(c1nc(C)c(C)s1)=O C1(C(=O)OC)N(C(=O)CC2CCCN2C)CCC1(C)C N1(C(C(CC2CN(C(C3C(C)CCOC3)=O)C2)F)=O)CCC(F)(F)C(F)C1 c1(CC(C(=O)NC(CC)CNC(c2ccn(C(C)(C)C)n2)=O)=O)ccc(F)cc1 C1(CNC(c2c(C)ncn2O)=O)CN(C(C2CC(C#N)C2)=O)CC(C(F)(F)F)O1 C(N=c1[nH]c(=NCCC(=O)N2CCCC2)[nH]c2c1CCCCC2)c1n(C)ncc1Cl C1(C#CC(=O)N(CC(=O)NCCC2CCCN(C)C2)C2CC2)(CC)COC1 CC1CC(C(=O)NC(C)C(C)F)N(C(=O)CCc2nncs2)C1 C1(N(CCOC)C)CCN(C(=O)C(C)NC(=O)COc2cccc(OC)c2)CC1 c1(OC)ccc(C(N)=O)cc1NC(c1nc(Br)cs1)c1nnnn1CCC1CC1 N1(C(c2n(C)c(=O)ccc2)=O)CCCC12CCC(NC(=O)Cc1cc[nH]n1)CC2 c1(OCC)ccc(Nc2oc(C)nc2C(N2CCC(C(N)=O)C2)=O)cc1[N+](=O)[O-] CC12CC(C(=O)NC3CC3c3ccc([N+](=O)[O-])cc3)(C1)C1(CCOCC1)O2 C1(CNC(c2cn(CC)nn2)=O)CN(C)CCN1C(=O)CCc1ccccc1F CCCC(C(=O)NOC(C)C)NC(c1cccc(=O)n1C)=O C1(NC(COCC(=C)C)=O)CCCC12CN(C(=O)C(c1ccc(C)cc1)C)C2 O=C(CCN=C(NCCF)N1CCC2(CCOCC2)C1)N1CCOCC1 C1(NC(=O)CCc2ccc[nH]2)CC2(C1)CC2C(=O)NC1(CF)CCCC1 C(C)(CS(C)(=O)=O)NC(CCN(C(=O)Cc1cnn(C)c1)CC)=O c1(C(N2CCC(CNC(CCC(C)OC)=O)CC2C)=O)c[nH]c2cc(Cl)ccc12 C1(NC(CC(CNC(=O)Cc2cccnc2C)OC)=O)CC2CC1OC(=O)N2 CCC(CC(=O)N1CCCC1CNC(=O)CSCC)CC(C)C C12(CN3C(C)(C)C(NCc4ccccc4)CC3)CNCC(=O)N1CCOC2 c1(CC(=O)NC2CC(C(=O)NCCCC#C)C2)cccc(F)c1 C(=O)(CCC(C)(F)F)NC(C)C(=O)NOC1CCC(O)C1O CC1CCCc2cc(C(=O)NCCCNC(C34CC(C)(C3)OC43CCC3)=O)nn21 C12(C(N(CC(C)(C)O)CC(C)(C)O)=O)CCC(CN(Cc3cc(Cl)ccn3)C1)C2 c1(OCCC(=O)NC(CCCNC(C(C)C#N)=O)C)ccc(C(C)(C)C)cc1 CC1(C)CN(C(=O)CCF)CC2(CN(C(c3ccc(=N)[nH]c3Cl)=O)C2)O1 c1(CC(=O)NC2(CNC(CCOCC#C)=O)CC2)ncn2c1CCCC2 N1(C(C(C)OC)=O)CC2(COC(CNC(=O)COc3ccc(Cl)c(Cl)c3)C2)C1 C1(CC)CN(C(c2c(C)cccc2F)=O)CCN1C(=O)COc1cccnc1 Cc1cc(-c2nc(-c3cncs3)nn2C2CCOC(C)C2)nc(N2CCCC2)n1 c1(C(C(=O)NC)N(c2ccccc2)Cc2ccn(C)n2)cnn(CCO)c1 C1(C(=O)NCCN(C(=O)CN(S(C)(=O)=O)C)CC)CC(C(C)(C)C)=NO1 N1(C(C(CC)(C)O)=O)CCCC(NC(c2c(C(F)(F)F)noc2C(C)C)=O)CC1 N1(C(CCCOCC=C)=O)CC(C)OC2(CCN(C(=O)C(C3CC3)SC)C2)C1 C1(C)(CNC(C(CC#C)C2CC2)=O)CN(C(c2nc(C3CC3)cs2)=O)C(C)(C)C1 C1(NC(=O)C(N2CCC(C3CCCN3C(=O)C(F)CC3CC3)C2)=O)CCOCC1 c1(C(=O)NCC(CC(C)C)NC(=O)COC2CC2)cc(=O)n(C)c2ccccc12 c1(C(=O)NCC(CC=C)NC(=O)C(C)(F)CC2CCCC2)cn2ncccc2n1 c1(NS(C)(=O)=O)nc(CC(=O)NCC2C(C(=O)NC3(CF)CCC3)C2)cs1 c1(C(=O)NC(c2ccc(Br)cc2)C2C(C(=O)OC)C2)cccc(=O)n1O N1(C(c2c(C)ccs2)=O)CCC2(CC(NC(C3CC34CC(F)(F)C4)=O)C2)C1 c1(C(=O)NC(c2cn(CCCC)nn2)(C)C)ccc(C(C)(C)C)cc1 C1(N(C(=O)COCC2CC2)C(C2CCC2)C)CCCCO1 C(=O)(CN(C)C(C1(CC)CC1)=O)NCC1(CCOCC)CC1 N12CCN(CC1)CCC1(CC1)C2=O.c1(C(C(=O)OC)=O)cscc1Br Cc1cc(Cl)c(C(=O)NC(C)CNC(=O)C(C)(C)C(C)O)cc1[N+](=O)[O-] c1(C(N(CCNC(c2c(O)ccc(C(=O)OC)c2)=O)C)=O)cccc2ncnn12 CCC(CC)(CCNC(=O)CS(=O)(=O)NC)NC(c1ccc[nH]1)=O CC1CN(C(C23COCC2C3)=O)CCN1C(=O)Cc1ccc(O)cc1Cl c1(CC(=O)NC(CC)CN(C)C(c2cscc2Cl)=O)ccnnc1O C1(CC(N2C(CNC(CC3N(C)CCCC3)=O)CCC2)=O)CCC(C)(C)CO1 Cc1cc(C)c(C#N)c(NC(=O)C(N2CCN(C3CCCC3)CC2)=O)n1 C1(C(=O)NCC2=CCN(c3c(C)c(Cl)ncn3)CC2)CCc2nnnn2C1 C1(NC(CCSC)=O)CC(NC(c2c[nH]c(C(F)(F)F)c2)=O)C12CCC2 N1(CCNC(C2C(COC)C2)=O)CCCN(C(=O)C(F)CC2CCOC2)CC1 C1(O)(CNC(c2cc(C(F)(F)F)on2)=O)CCN(C(C2CCCS2)=O)CC1 C1(CCNC(c2n(CC=C)ccc2)=O)CN(C(c2cc(=O)cc[nH]2)=O)CC(C)O1 c1(C(=O)NC2CC(CNC(CC3C(C)=NN(C)C3=O)=O)C2)n[nH]c2cccnc12 c12cc(nc(CO)n1)N2.N1(C(c2cnccn2)C)CCN(CC2CC2(C)C)CC1 c1(C(=O)NC2CC(C)N(C(=O)C=C3CC3)CC2)cc2c(cc1Cl)OCO2 c1(C(=O)NC2CCC(C)(NC(CC3N(C)CCC3)=O)CC2)nc[nH]c2ncnc1-2 C1(F)(CNC(C2(C(=O)NC)CCC2)=O)CC(NC(=O)CC2C=CCC2)C1 C1(NC(c2csc([N+](=O)[O-])c2)=O)CC2CCC1N2C(C1(F)CCC1)=O Cc1nc2ccc(C(=O)NCC#CCNC(C3(C)CCCS3(=O)=O)=O)cc2s1 N1(C(COCC#C)=O)CCN(C(c2cn(C3CC3)nn2)=O)CC1CC(F)F C(=O)(C#CC1CCCO1)NCCC(CC)(CC)NC(=O)Cc1ccc(OC)cc1 C#Cc1ccc(Cl)c(C(=O)NCC(O)CNC(=O)C(F)C2CCC2)c1 C(=O)(C(C)(C)CC(C)C)N1CCCC(NC(COCc2cccc(OC)c2)=O)C1 CC1(CNC(=O)CCc2ccccc2O)CC(F)(F)CN1C(=O)C=CC1CCC1 C1(C(=O)NCC2(C)C(C)CN(C(=O)Cn3ccnn3)C2)CCCN2CCCCC12 c1(C2CC(N)C2)ccccc1F.n1(CC)cc(CCCNC(C2CCNC2=O)=O)nn1 Cc1cc(F)ccc1C1(C(=O)N(CC(O)CNC(c2ccc(F)cc2)=O)C)CC1 c1(C(N(C)CC2(CNC(COCCOC)=O)CC2)=O)noc2c1CC(C)CC2 c1(C(=O)OCC)cnc(C(N2CCN(CCC3CC3)CC2)C(=O)NCC)nc1 c1(C(=O)NC(C(C)NC(c2cc(F)ccc2F)=O)C)cn(C)c2ncccc12 C12(NC(C3CC(OCC)C3)=O)CCCC1CN(C(=O)C(C)(C)N(C)C)C2 C1(C(=O)NCCC(C)N(C(C(CC)OC2CCCC2)=O)C)(C(=O)OC)CC=CCC1 C1(NC(CSCCN(C)C)=O)CCCC(NC(c2cc(C3CC3)no2)=O)CC1 c1(C(=O)NC2C(NC(C3(CC)CC3(F)F)=O)CCCC2)ccc2n[nH]c(C)c2c1 c1(OC)ccc(I)c(CCC(=O)NC2CCCN2C(C)C)c1.C12CCN(CC1)C2 c1(C(N2CC(CC(C)NC(=O)CCSC(F)(F)F)C2)=O)cnc2ccccc2n1 C1(NC(c2ccncc2Br)=O)CC2CC(C1)N(C(C1CC(F)(CO)C1)=O)C2 n1(CC)cc(Cl)c(C(N2CCC(Cn3cc(CN(C)C(C)=O)nn3)C2)=O)n1 C1(NC(c2ncn(CC)c2)=O)CC2CC(C1)N(C(=O)C(C)(C)c1cccnc1)C2 N1(C(C2CC(CCC)OCC2)=O)CCC(NC(=O)CC#N)C(C(N)=O)C1 c1(CC)oc(C(=O)NC2CC(C)N(C(c3cn(CCF)nn3)=O)C2)cc1C Cc1cc[nH]c(=N)c1C(N1CCN(C)C(CNC(C2(Cl)CC2(F)F)=O)C1)=O N1(C(C=Cc2cncc(C)c2)=O)CC(NC(=O)C(C)(C)CO)C2CCCCC12 C(c1sccc1Br)=CC(N1C(CNC(C2CCN(CC)C2)=O)CC1)=O CC1(NC(=O)CSc2ccc(Cl)cc2)CCCN(C(=O)CC2CCCO2)C1 N1(C(c2c(C(C)(C)C)ccnc2)=O)CCCCC(NC(=O)CN2CC3CC3C2)C1 CC1CC(=O)CCN1C(=O)C(C(C)(C)C)n1cc(Br)cn1 c1(C(=O)NC2CCCCC2(F)F)cnc2c(C3=CCCCC3)cnn2c1 C1(C(=O)NCC2(C(=O)NCc3cc(CO)[nH]n3)CC2)COCCOC1 CC1CC=CCC1C(=O)N(CCCNC(=O)C(c1cccc(Cl)c1)O)C1CC1 Cc1ccc(C(CNC(C2CCC(=O)N2C)=O)NC(=O)CNC=O)cc1 c1(C(N2CC(NC(C3(CC=C)CC=CC3)=O)C3C2C3)=O)ccc(S(N)(=O)=O)cc1F c1(C(N2CCN(C(C3C(OCC)C3C)=O)C(C(C)C)C2)=O)ccnc2ccnn12 Cc1ccc(C(N2CC3C(CN(C(=O)CNS(=O)(=O)C4CC4)C)C3C2)=O)c(N)n1 c1(C(N2Cc3cncnc3C2)=O)nc2ccc(-c3ccc(CN4CCC4)o3)cc2o1 c1(NCC(CN(C)C(=O)OC(C)(C)C)CO)cn(C)[nH]c1=NC(=O)OC(C)(C)C N1(C(CN(C)CCO)=O)CC2CCC1C(CNC(C1(C)CC(O)CN1C)=O)C2 C1(c2nnnn2C2COC2)(NCCC2(C)CC2)CC2(CCCNC2=O)C1 c1(C(=O)NCC2N(C(C(C)Cc3ccco3)=O)C3C(C2)C3)ccc2cnoc2c1 N1(C(C2C(CC)OCC2)=O)CCC(F)(F)C(CNC(C23CCC(CC2)CO3)=O)C1 CC1CCN(C(c2nscc2Br)=O)C1CNC(c1cnnn1C1CC1)=O Cc1ccc(F)c(C(=O)NCC2(C)CN(C(c3c(C)ncn3C)=O)C2)c1 CC1(C(N2CCOC3(C2)CN(C(C2CC(O)C2)=O)C3)=O)C2Cc3ccccc3C12 c1(OC)ccc(S(=O)(=O)NCCOC2CCCNC2)c2ccccc12 NS(=O)(=O)CCCCCCCCC(=O)N1CC(NC(=O)C=CCF)CC2(CC2)C1 CCCC(C)CC(=O)N1CC(CNC(c2cnc3n2CCS3)=O)C(C)(C)C1 c1(C(N2CC(C)(NC(C(C(C)(C)C)OC)=O)C2)=O)cc(C)cc(C)c1O C12(C(=O)NC(C(C)NC(C3CCC3c3nc(S)n[nH]3)=O)C)CCC(=O)N1CCS2 CC1C(C(=O)NCC2CN(C(c3cnn(CC4CCC4)c3)=O)C2)C(O)C(=O)N1C c1(C(N2C(CNC(c3c(CC)nco3)=O)CCC2)=O)ccc(C(F)F)c(OC)c1 c1(N2CCCC(NC(C=COCC)=O)C2C)nn2cc(C)nc2s1 C(=O)(CCCN(C)N=O)NC(CCCNC(C1CCN(S(CC)(=O)=O)CC1)=O)C N1(C(C2CC(C)(CC)C2)=O)CCOC(C(C)NC(c2cnc(C)[nH]2)=O)C1 CC1CCN(C(c2cccn2C)=O)CC1CNC(=O)CNC(c1cscn1)=O c1(C(C)C)nccc(C(N2CCCCC2C2(NC(=O)CC3CCCO3)CC2)=O)n1 n1(CC)nc(C(C)C)cc1C(=O)NC1CCC1CNC(=O)CC(C)OC c1(C(N(C(C)CNC(=O)CCC2CCN(C)C2)C)=O)cn(C)c2ccccc12 CN1CC(NC(=O)CNC(=O)CCS(C)(=O)=O)C(C)(C)C1 N1(C(C(C)OCC#C)=O)CCN(C(=O)C=Cc2cncs2)C(c2ccncc2)C1 N1(C(C(C)SC(F)(F)F)=O)CCC(O)(CCNC(c2ccsc2Cl)=O)C1 c1(C(N(CCCNC(C(CC(C)C)NC(C)=O)=O)C)=O)cnc2ccccc2c1 C1(NC(CCC2(NC(C(COC)C)=O)CCCC2)=O)CCN2CCCCC12 c1(C(=O)OC)cc(C(=O)N(CC(C)(C)CNC(=O)C(O)C2CCC2)C)c(F)cn1 C(C)(CNC(=O)C(C)CC)(CC(C)C)NC(c1cc(CCC)nn1C)=O c1(OC)cc(F)c(C(N2CC(CNC(c3ccco3)=O)C3CC23)=O)cc1OC C1(O)(CN(C)C(C2CSCN2C)=O)CCN(C(c2cscc2Cl)=O)CC1 CC1(C)CCCC1CNC(C1CCC1NC(=O)C1=C(Cl)CC1)=O C1(OCC)CN(C(=O)OC)CCN1C(c1ccccc1Cl)C(=O)OC N1(C(C(C(=C)C)(C)C)=O)CC2(CC(NC(c3cccc(F)c3SC)=O)CO2)C1 c1(COC)ccnc(C(N2CCN(C(=O)CSc3nncn3C3CC3)CC2)=O)c1 C1(C(C)(C)C)(CN(C)C(c2ccc(F)cc2)=O)CCN(C(C2CC(O)C2)=O)C1 C(C(=O)NC(CCN(C(=O)CCn1cncn1)C)C(C)C)(C(C)C)OCC(C)C C1(C(=O)NCCC2(OC)CN(C(C=C(CCC)C)=O)C2)CC12CCCC2 Cc1[nH]nc(Cl)c1C(N1CCC(C2CCCN2Cc2nc(O)n[nH]2)CC1)=O N(C1CCCc2cc(NC(=S)N)ccc21)S(c1c(C#N)ccs1)(=O)=O C1(CC(=O)NCC(C)(C2CC2)OC)C2CN(C(c3nc(=N)cc[nH]3)=O)CC12 C1(C#N)(C(=O)NC2CN(C(CC3ON=C(CC)C3)=O)C2)CC2(CCC2)C1 Cc1nc(C2CC2)nc(O)c1C(=O)NCC1CC(NC(=O)C(Cl)=CCl)C1 c1(C(N(CC(=O)NC(C)CC2CCC2)CC2CC2)=O)cnccn1 C1(CC)C(NC(c2cc(SC)c(C)o2)=O)CCN1C(=O)Cc1csc(S)n1 CP(C)(=O)c1c(NC(N2CCCC(n3ccc(C(F)(F)F)n3)C2)=O)cccc1F C1(CNC(C(C)OC)=O)CC2(CC(NC(=O)C(C)Cc3ccc(F)cc3)C2)C1 N1(C(C(c2ccn(C)n2)C)=O)CCC(C(C)(C)NC(=O)C=CC(F)(F)F)C1 c1(OC)cnc(F)c(C(N2CC3CC3(CNC(=O)C=CC(=O)NC3CC3)C2)=O)c1 CC1(C)CC(NC(=O)Cc2ccsc2)CCN(C(C2CCCC3(CCC3)C2)=O)C1 CS(=O)(=NC(=O)c1ncn(-c2ccccc2)n1)c1ccccn1 C(=O)(C1=CCC(C)CC1)NCC1N(C(CC2(COC)CCCC2)=O)CCC1 CC(C(=O)NC(C)(C)CCCNC(C1CC(=C2CC2)C1)=O)C(C)n1cccn1 CCCC(C)CC(=O)NC12CCCC(NC(=O)CC(CC)SC)(C1)C2 CC1CCCCN1C(c1ccc(NC2CC2C(=O)NCC(N)=O)cc1)=O n1(CC)cnc(C(=O)NC(CC2CC2)C(=O)NCc2nc(C(C)C)n[nH]2)c1 c1(CC(C(=O)NCCOC)NC(c2scnc2Cl)=O)ccc(Cl)cc1Cl c1(C(=O)NC2CN(C(c3ccc(O)cc3)=O)CC2F)cc(Cl)cc([N+](=O)[O-])c1Cl C1(C(=O)NC2C(NC(=O)CCC3CCCCO3)CCC2)CCn2c(O)nnc2C1 c1(C(=O)NC(C(C)C)C(C)C)n[nH]c2c1CN(C(=O)CCCN(C)C)C2 C(C(=O)NC1CN(C(=O)CC(C)(C)C)CC1C(F)F)(C(C)(C)C)SC c1(CC(N2C(CN(C(C(C3CC3)OC)=O)C)CCC2)=O)noc2ccccc12 C1(NC(Cc2c(S(C)=O)cccc2)=O)CCN(c2nccnc2F)CC12CCC2 C12CCN(CC1)C(=O)Cc1ncc(s1)C(=O)N2.C1(C(=O)OC)(COC)CCCO1 c1(CNC(CCCSC)=O)c(C)nn2c1CN(C(=O)CC1CC3(CC3)CO1)CC2 C=CC1CN(C(=O)OC(C)(C)C)CC1C(N1CCCC1c1cncn1C)=O N1(C(CC=C=C)=O)CCC(NC(c2cc(Cl)ccc2C)=O)C(CO)CC1 CCC(CC)CCCC(=O)NCC1(NC(=O)CCCOC(C)C)CCOCC1 N1(C(c2cn(C(C)C)nc2)=O)CCC(NC(=O)Cc2ccc(F)cn2)C1(C)C c1(OC)ncc(C)c(C(=O)NCC2CN(C(=O)CCN3CCC(O)CC3)C2)c1Cl Cc1ccc(NC(=O)CC2(C)CCN2C(=O)CC2COCC2O)cc1O CC1(C)CC(C(=O)NC2(c3ncccc3F)CC2)CCN1C(C1CCC1)=O C12(C(=O)NC(CNC(c3ccc(CC)nc3C)=O)C)CCC(N(C)C)(CC1)CC2 CC1CN2CCN1CC2C(=O)NCC1(NC(c2cnc3ncccn23)=O)CCC1 C1(COC)CC(NCc2cnn(C)c2)CN1C(=O)OC(C)(C)C N#CC1(C(=O)NC2CC(CCNC(C=CC(=O)NN3CCCC3)=O)C2)CCOC1 c1(C(=O)NC2C(NC(=O)Cc3cnccn3)C2)ccc(F)c(CO)c1 O=C1CCN(Cc2ccccc2)C(=O)N1CCCc1cc(CC2CCOC2)no1 c1(C(=O)NCCN(C(Cc2c(C)nsc2)=O)C2CC2)ccn2ncc(C)c2n1 CCCC(O)CC(=O)N1CCC(C)C(CNC(c2c[nH]c(C)c2)=O)C1 c1(C(N(CC(=O)N(CCN=[N+]=[N-])CC)C)=O)c(Cl)cnn1C C1(NC(CCC2(C#N)CCC2)=O)CCCN(C2CC2)C1 C(=O)(C1=CC(C)(C)C1)NCC(CC1CN(C(C(C)OCC2CCOCC2)=O)C1)(C)C N1CC(C)(C)CC1.c1(CNC(C)=O)nc(C)c(C(=O)O)o1 C(CS(=O)(=O)CC(=O)NC(C1(O)CN(C(C2CC3(C2)CC(C)C3)=O)C1)C)OC c1(NC2CC3OC(=O)OC3C2)cccc(S(F)(F)(F)(F)F)c1 c1(C(C(N2CC(C(C)(C)O)OCC2)=O)=O)ccc2c(c1)CCC2 c1(NC(C2N(S(c3cn(CC)nc3)(=O)=O)CC(C)C2)=O)cc(C)c(Br)c(F)c1 c1(CC)ccc(C(N2CCC(CNC(=O)Cc3c[nH]nc3C)(OC)C2)=O)cc1F C1(NC(C(C)Cc2ccccn2)=O)CN(C(c2cc(CO)on2)=O)CC(F)(F)C1 c1(C(=O)OC(C)(C)C)cnc2c(c1)CCCO2.N12CCC(C)C1CNC(C)C2=O c1(CCC)cc(C(=O)N(CC(O)CNC(=O)CNC(=O)CC)C)n[nH]1 N1(C(C(C(C)CNC(C2CCCCCC2)=O)F)=O)CC2C3CCC(C3)C12 c1(CC)nn(C)cc1C(=O)NC1CCN(C(=O)CC2CCC(=O)CC2)C1C C1(C(=O)NCC(C)(C)NC(=O)CCN2CCCCCC2)(CO)CCCCC1 C1(NC(CCCOC(C)C)=O)CC(NC(=O)CC2(C#N)CCCCC2)C12CCC2 C1(C(N2CC(CC(C)NC(=O)CC(C)(C)O)C2)=O)CC(=O)N(C2CCCCC2)C1 c1(C(=O)NCC2CN(C(C(C)(C3CC3)OC)=O)CC2O)cc(C#N)c(F)cc1F C1(CNC(CC=CCC)=O)C(CNC(=O)CN(C)CCOC)C1(F)F N1(C(Cn2ncc(C#N)c2)=O)CCC2CN(C(c3ccoc3Cl)=O)CC2C1 N1(C(C=CC=CC)=O)C2CCC1CC(O)(CNC(c1cn(CCCF)nn1)=O)C2 c1(OC)ccccc1-n1nnnc1C1(NC(COC)CC(C)C)CCC1CC#N Cn1ccc2cc(C(N3CC4=C(C3)CN(C(C3CCCC35CC5)=O)C4)=O)cnc12 Cn1ccc(C2(C(=O)NCCCN(C(=O)C(O)Cc3cnc[nH]3)C3CC3)CC2)n1 C(=O)(C(C)(C)C(F)F)NC(C)CCNC(c1ccncc1Cl)=O N1(C(c2n(C(CC)C)ncc2)=O)CC(C(F)(F)F)C(CNC(=O)COC(C)C)C1 N1(C(c2cc(C)nn2C2CCC2)=O)CCC(O)(C(C)NC(C2CCCO2)=O)CC1 C(=O)(CCCCCF)NC1CC(O)(CNC(c2ccc(N(C(C)=O)C)cc2)=O)C1 Cc1ccc(CC(=O)NC2(CNC(C3C=CC=CC=C3)=O)CCOCC2)c(Cl)c1 N1(CCC(=O)N(C)CCOCCN(C)C(C2CSCCS2)=O)CCCC1=O N1(C(C2C(=C)C2)=O)CCC(CNC(=O)CC2=CCCCC2)C(F)(F)CC1 N1(C(c2c(C)ccs2)=O)CC(C)C(NC(C2CC3(CC3)C2)=O)C(C)C1 CC(C)C(C(=O)NCCCn1ccnc1)NC(C1CC2CC2C1)=O c1(C(N2C(C)CC(CNC(c3cnc(S)nc3)=O)CC2)=O)cc([N+](=O)[O-])nn1C c1(OC)ccc2c(n1)NC(C(=O)NC(C)(C)CNC(C1(Cl)CC1)=O)C2 c1(C(C(=O)NC2CCN(C(C(CCSC)O)=O)C2)(C)C)ccc(F)c(F)c1 C1(CNC(=O)CCOCC2CCCO2)CCCCC1NC(=O)C(F)(F)C1CC1 c1(NCC(=O)NC2N(C(CC3(C)CC3(Cl)Cl)=O)CC2)ccccc1C(N)=O N1(C(c2cncc(C#N)c2)=O)CCC2(CCC2)C(NC(c2ccccc2F)=O)C1 C1(C(=O)NC(CNC(COCC(=O)NC)=O)C)CCCC1CF Cc1[nH]nc(C(=O)NC(C2CCCN(C(=O)CCCc3cncs3)C2)C)c1Cl N1(C(CC=CC=C)=O)CCC(CCC(=O)NCc2ccc(Cl)o2)C1 c1(COC)cc[nH]c1C(=O)N(CCC(=O)NC(c1cccnc1)CO)C(C)C CC(C)CC(C)(CNC(=O)Cc1sc(O)nc1O)NC(C1CC2CCC1CC2)=O c1(C(N2CC(C)C(NC(=O)CCC3CCCN3C)C2)=O)cnn2c1C(=O)NCC2 Cc1cc(C(N2CC(NC(=O)CCOC3CCN(C)CC3)C(C)C2)=O)cc(C)n1 C#CC1(O)CC(C(=O)NC(C2CCCC2)CNc2ccc(CC=C(C)C)cn2)C1 CCC(C(=O)NCC(C)(Cn1cccn1)NC(=O)CCC(C)C)C(C)(F)F c1(NC(=O)CC(CC2CC2)NC(=O)C(C2CC2)C2CC2)cnc(O)c(F)c1 c1(OC)ccc(NC(=O)CCOC(CNC(C2OC3CCC2C3)=O)CO)cc1F N1(C(c2c(C)nc(Cl)cc2)=O)CCC2(CC(C(=O)NC3CSC3)=NO2)C1 C1(c2cn(C)nc2)CC(N=c2cccc(S(=O)(=O)NCC3CCCS3)[nH]2)CCO1 c1(C(C)(C)C(=O)NC2CCC(NC(=O)CSCC(N)=O)C2)cccc(F)c1 C1(C#CC(=O)NC2(CO)CCCN(C(C3(F)CCS(=O)(=O)C3)=O)C2)(CC)COC1 CCC(C)C(C)(O)CNC(C1C=CCN1C(=O)CC1(C)CCOC1)=O C(CNC(C1(F)CC=CC1)=O)(C(=O)N1CCC(OC(C)C)C1)OC N1(C(=O)CCc2nc[nH]n2)CCOC(CC(N2CCC(CF)C2)=O)C1 N1(C(C2CN(C)C(=O)N2)=O)CC2OCC(NC(=O)CCCc3cccnc3)C2C1 C1(C(=O)NCC2CCC(CO)CC2)CC2CCC1N2C(c1c(F)cncc1F)=O N1(C(c2c(C)cncc2)=O)CCN(C(C2CCC(F)(F)CC2)=O)C(C)CC1C C(=O)(C#CC1(C)CCCO1)NCC1(F)CC(NC(CC(C)c2cnn(C)c2)=O)C1 c1(C(=O)NC23CN(C(C4CC(=O)NCC4)=O)C(C2)C3)cc2n(c1)CCC2 N1(CCCC)CCCCC1C(=O)NCC(C)N(C(=O)CC(C)F)CC c1(N(C)CC2N(C(CSCC#C)=O)CCCC2)nc(CC)nc2sccc12 N1(Cc2nnc(CCC)s2)C2CCCC1CN(C(=O)C(C)OCOC)C2 N1(C(CCSC)=O)CCN(C(c2nc(O)sc2C)=O)C(c2cccc(Cl)c2)C1 c1(C(=O)NCc2nc(C)on2)ncccc1NC(=O)Cc1ccsc1 CC1=C(C(=O)NCC2CC2CNC(=O)Cc2c[nH]nc2O)CCCC1 C1(C(N(C2C(OC)COC2)C)=O)C2CN(C(=O)CCc3nccs3)CC12 N1(C(c2cc(CC(C)C)nn2C)=O)CCN(C(C2(C)CCC2)=O)CC1C(F)F C1(CC=C)(C(N2CC(F)C(F)C2)=O)CCN(C(c2ccc[nH]2)=O)C1 N1(C(c2c(C)cc(F)s2)=O)CCCC(N(C)C(C2(C(F)F)CC2)=O)CC1 CCC(CC)(CC)C(=O)N1CCC(O)(CNC(c2c(C)cc(=O)oc2C)=O)C1 n1(C(C)CNC(=O)CCn2cc(S(N)(=O)=O)cn2)cc(C(=O)O)c(O)nc1=O c1(OC)cnc[nH]c1=NCC1(C(C)(C)C)CCN(C(=O)CN2CC3CCC2C3)C1 C1(CNC(C2CCC23CCC3)=O)CC(F)(F)CN1C(C12CCCC(C1)OC2)=O CC1(C(=O)NC2CCC(CNC(=O)Cc3ncc(F)cc3F)C2)CCCC1(F)F C1(C(N2CCCC(=C)C2)=O)CCN(C(C2(C(=O)OC)CC2)=O)CC1O C(=O)(C1=CCS(=O)(=O)C1)NC1C(NC(c2cnc(=N)[nH]c2)=O)CCCC1 CC(CC(C)C(F)F)NC(C12COC(C1)C(NC(=O)CCc1nc(O)n[nH]1)C2)=O c1(CC)nc(C)ncc1C(=O)NC1CCCC(NC(=O)Cn2cncn2)CC1 c1(-n2c(C(=O)NC3C(CNC(C4(CCC)CCC4)=O)C3)cnc2)ccccc1C N1(C(C(COCC)NC(=O)Cc2ccsc2C)=O)CC(C)C1(C)C N1(C(Cc2ncc(C)s2)=O)CCOC(CN(C)C(C2CC(F)C2)=O)C1 c1(C(C(=O)NCC(CC)NC(C2(C)C=CCCC2)=O)(F)F)ccc(C)cc1 C(=O)(CC1=CCCC1)NCc1c(CNC(=O)CC2CCOC2)cco1 C(c1cc(F)c(F)c(F)c1)=CCC(=O)NOCC(=O)NC1(C(=O)O)CCC1 Cc1ncc(NC(C2(C)CCN2C(=O)CC2CCC(C)(C)CC2)=O)cc1Br C1(NC(C2(CCC)CC2)=O)CCCCCC1NC(=O)Cc1ncn(C)c1C c1(N2CCC(C)(CCC)C2)ncnc(NC2CCC(C)(C)C2)c1C Nc1cc(C(N2CCCC(F)(CNC(=O)C(O)Cc3cnc[nH]3)C2)=O)ccc1Cl C=CCCN=C(NCCN1CCC(C)CC1)NCc1cccc(C)c1 C1(CC)CN(C(=O)OC(C)(C)C)C(C)(CSc2snnc2-c2ccc(F)cc2)C1 N1(C(C2C3CCN(C(C(C=C)OC)=O)CC32)=O)CCn2cnnc2C1C C1(NC(CC(CC)SC)=O)CCN(C(=O)CN2CCCNC2=O)C(C)C1 Cc1nn2cccnc2c1C(N1CCC(C)(CNC(=O)C(F)=CC2CC2)C1)=O c1(C(=O)NC(CNC(Cc2ccc(OC)cn2)=O)C2CC2)c(F)ccc(F)c1Cl Cc1c(Cl)ccnc1C(N1CCCC(CCNC(=O)C(C(C)O)N(C)C)C1)=O C1(CCOC)CN(C(c2ccnn2C2CC2(F)F)=O)CCN1C(=O)C1CC1 CON1CCC(C(N2CCC(C(C)NC(c3cc(Br)n(C)n3)=O)C2)=O)CC1 c1(CCC)cc(C(N2CCCCC2C2(NC(=O)C(F)=C3CCC3)CC2)=O)ccn1 c1(C(N2CCCC(CNC(c3cc(CN(C)C)on3)=O)C2)=O)nccc(Cl)c1O c1(C(=O)NCC2(C)CCC(NC(CCOCCC)=O)C2)cccc2[nH]c(=N)oc12 CC1(C)CCc2oc(C(NC3=COCCC3)=O)cc2C1=O C12(C(N3CC(CCNC(C4(F)CC(C(=O)OCC)C4)=O)C3)=O)CCN(CC1)CC2 CCCCCS(=O)(=O)CC(=O)N1CCCC1CN(C(=O)CN(C)CC)C1CC1 CC1(NC(=O)CC(O)Cc2ccccc2)CCN(C(=O)Cn2nnc(=N)[nH]2)CC1 c1(CC)cc(F)ccc1C(=O)NC1CC(NC(C2COC(C)C2)=O)C1 c1(CC(=O)NC2C(CO)CCN(C(C=CCC)=O)C2)c(C)cc(C#N)cc1C c1(CNCC23C(CN(C(Cc4cc(C)ncc4)=O)C2)C3)cnc(F)c(C)c1 Cc1cccc(NC(C2CC3CC3N2C(c2cc[n+]([O-])cc2)=O)=O)n1 CC1(C)CN(C(c2cc3n(n2)CCC3)=O)CCC1NC(=O)C(C#N)C1CC1 c1(NC(C2(CN)CC2)=O)cc(C(F)F)ccc1COC(c1cccc(F)c1)=O c1(-n2c(C3C(C)(CC)C3)nc(-c3ccn(C)n3)n2)cc(Cl)ccc1C Cc1c(C(N2CC(C)(NC(C3CCC=CO3)=O)C2)=O)cncc1Cl c1(C(=O)NC23CC(CN=c4nc(SC)[nH]s4)(OC2)C3)ccc2cnnn2c1 c1(CO)cc(Cl)ccc1OC1CC1(F)C(=O)NC1(OCC)CCC1.C1(=O)CCN1 c1(CN2CCC(C(N(CCS(C)(=O)=O)C(C)C)=O)C2)c(Cl)cc(Cl)cc1Cl c1(SCC)cc(C(=O)NCC(C(C)C)NC(=O)CC2(C)CC2(F)Cl)ccn1 C1(CC)C(NC(=O)CCCN=[N+]=[N-])CCCN1C(C1CCCCS1)=O c1(OC)cnncc1C(=O)NCCn1ccc(C(=O)Nc2cnn(C)c2C(N)=O)c1 C1(C(N(CCC(=O)OC)CC)=O)CN(C(c2cnnn2C2CC2)=O)CC1CC c1(C(=O)NCC(C(C)C)NC(=O)CC2CN(C)C2)cc2cc(Cl)sc2[nH]1 O(NC(=O)C(CCC1CC1)NC(=O)CCc1ccsc1)CC(=C)C c1(C(C)(C)C)ccc(C(=O)C(=O)NCCOC2CCN(C(=O)CCF)CC2)cc1 CCC(CCCC(=O)NCC1CC(SC)C1)NC(=O)CN(C1CCCC1)C CN1CCCC(NC(=O)C(C)(C)C2CCCN2C(=O)C(C)(C)C(F)F)CC1 n1(CC)ccc(C(N2CC(CC(=O)NC3CCCC3CCO)CC2C)=O)c1C CCCCS(=O)(=O)CC(=O)NC(C)(CNC(=O)C(C)OC)C(C)C C(=O)(C(C)C(C)C(C)(C)C)NCC12N(C(C3(C#C)CCCC3)=O)C(CC1)CC2 N1(C(C#C)C2CC2)CCN(CC(c2cc(C(C)C)cs2)O)CC1 C1(NC(Cc2c(C)con2)=O)CN(C(c2nnc(O)cc2O)=O)CCC12CCC2 N1(CCOC)CCCCCC1CC(C)C.C12CN(C1)C(=O)COCCO2 N1(C(CNC(=O)NC)=O)C2CCC(C2)C1C(=O)NCc1cc(C)ns1 C1(C(N(C2(C(=O)NC(C(F)(F)F)C3CC3)CCC2)C2CC2)=O)CCS(=O)CC1 N1(C(c2ccc(C(C)=O)c(F)c2)=O)CC2CCC(C1)N2C(C1CC=CCC1)=O N1(C(c2c(C)noc2C2CC2)=O)CCOCC(NC(=O)CC2(C)CCC2)C1 C1(NC(C(n2ncc(C)c2)C)=O)CCN(C(c2ncnc(C)c2C)=O)CC(O)C1 C=CCC(CNC(c1cc(C2CC2)ns1)=O)NC(c1c[nH]nc1OC)=O c1(C(N2CC(CC=C)(NC(c3ccc[nH]3)=O)C2)=O)cc2c(o1)CCCC2 C1(C(=O)NC2(C)CCN(C(Cc3cccc(C)c3)=O)CC2)CCC2CCC(=O)N12 C1(C(C)C)CC(C(N2CC(C(N)=O)(CNC(=O)C(C)(C)C#N)C2)=O)CCO1 N1(C(CC(C(C)C)NC(=O)C(C2CCOCC2)C)=O)CCC12CCN(C)C2 N1(C(C(c2ccco2)NC(CC=CC)=O)=O)CC(F)CC1CO C1(NC(c2cnc(C(C)C)[nH]2)=O)CC2CCC1CC2NC(c1ccc(=O)oc1)=O C(=O)(CC(O)C(C)(C)C)N(C1CCCCC1)CCNC(C1CCC(=C)CC1)=O C(CC(O)C(C)C)NC(c1ccc(C(=O)OC)o1)c1nnnn1C(C)C Nc1ccc(C(=O)NC2CC(O)CN(C(=O)Cn3ncc(Br)n3)C2)nc1N C1(OC)CC(CCNC(C2(OC)CC2)=O)N(C(=O)C(c2c(C)n[nH]c2C)C)C1 c1(CC)nnc(=NCCC(C)(C)NC(c2cnc3c(F)cccc3c2)=O)[nH]c1CC c1(C(N(CCC)CCNC(C2CCC2n2cccn2)=O)=O)c(N)sc(C)c1C C1(CCNC(C(CC)C)=O)CCCN(C(c2cc(C)n(C3CCCC3)n2)=O)C1 c1(C(=O)NC2CCN(C(C34C(C)OC(CO)(C3)C4)=O)CC2)cccc2nncn12 CC1(C(N2CCC(O)C(O)C2)=O)CCCN(Cc2ccc(Br)c(OC(F)F)c2)C1 N1(C(C(CC)N(C)C)=O)CCC(C)CC1CNC(C1(C)CC=CC1)=O CC(C)CCC(C(=O)NC1CN2CCC1(F)CC2)NC(C1CCOCC1)=O c1(C(N(C2C(N(C(CCCC)=O)C)CCCC2)C)=O)n[nH]c2c1CC1CC21 N(C)(S(=O)(=O)N1CCOC(CC(N)=O)C1)CC C(=O)(C(C)C(C)O)N(CCN(C(CN(C(c1c(C)occ1)=O)C(C)C)=O)C)C(C)C c1(C(=O)NC(CCCNC(C(c2scc(C)n2)C)=O)(C)C)coc(S(C)(=O)=O)c1 C1(NC(c2c(CC)onc2)=O)CCSC12CN(C(c1ccc3ncnn3c1)=O)C2 C(CNC(=O)C(C)(C)C1CCC1)(CC(=O)NCC1(F)CCC1)OC C1(NC(C(CSC)O)=O)CCCCC1CC(=O)NC1COCCOC1 C(=O)(C1CCCc2nn[nH]c21)N1CC2CC3C(NC(=O)Cc4cnoc4)C1C2C3 Cc1sc(C(=O)NC(C)CC(C)NC(=O)C(F)CC2CCC2)cc1[N+](=O)[O-] C1(C(=O)NCCc2cccc(F)n2)CCOCCN1C(C1OC2CCC1C2)=O c1(-c2n(C)ncc2)cn(C)c2ccccc12.c1nnnn1C1CC1.C1(=O)CN1 c12nc(cc(C)n1)CC1(CCC(=O)OC)CN2C1.c1(SCC(C)CO)ccccc1 n1(CC)nccc(NC(N2CCCSCC2C2CCC2)=O)c1=O CC(CNC(C1(CO)CCC1)=O)C(=O)NCCc1nncn1C C1(C(=O)NC2(CCN(C)C)CN(c3c(C)c(Cl)ncn3)C2)CCc2c[nH]nc2C1 C1(N(C(C(C)Oc2cccc(CC)c2)=O)C)CCCN(C(C2CSC2)=O)CC1 C(C)(C(=O)NCCCN(C(=O)CN1CCC1C)C1CC1)OCC CC(C(=O)NC1CC2C(NC(=O)CC3(n4cccn4)CC3)C2C1)C(F)F c1(COC(CCCNC(N(CC)CC)=O)=O)ccc(Oc2ccccc2F)cc1 Cc1ncsc1C(N1CCC(C(=O)NCCCc2cnccn2)C1)=O c1(C(=O)NC2C(C)C2)c(NC(=O)C(=O)c2ccco2)sc2c1CCCC2 c1(C(=O)NCC2CC3(CN(C(c4[nH]n(C)c(=O)n4)=O)C3)C2)cc2c([nH]1)CCOC2 C(CC(O)CO)N(C)C(C1(NC(=O)C(c2ccccc2)F)CC1(C)C)=O Cc1oc([N+](=O)[O-])cc1C(N1CCN(C(C2(F)CCOC2)=O)CC1CO)=O CCCCCCn1nnnc1C(c1cn(C)cn1)NC(C)C(=O)NCCF c1(CCCC=O)nc2ccccc2o1.N1(C(C)=O)CCN(C)C1=O c1(C(N2CCC(NC(C(COC)N(C)C)=O)C2)=O)nc(Br)n2ccccc12 CC1CCCC(OCC(=O)NC2CCN(C(=O)CN3CCNC(=O)C3)CC2)C1 C1(C(=O)NCc2onc(N(C)C)n2)C2CCN(C(=O)C(C)(O)C3CC3)CC12 c1(-c2nc(C)c(NC(c3c(C(F)(F)F)cccc3F)=O)s2)ccc2c(c1)CCO2 C1(CCC(=O)NC2CCN(C(=O)OCC)C2)CCCN(C(=O)CN(C)C(N)=O)C1 c1(NC(C2C(NC(c3ccc(SC)s3)=O)C2)=O)nc(O)c([N+](=O)[O-])c(O)n1 c1(C(=O)NC2(CN(C(C3(COC)CC3)=O)C)CC2)cccc(CC2CC2)c1Cl c1(C(=O)NC2CCC(C)N(c3nc4cccnc4s3)C2)ccc2ccccc2c1 c1(C(=O)NC(CNC(CC(C(C)C)C)=O)(C)C2CC2)nnc(O)c2c1CCCC2 N1(C(C2C(NC(C3CCC(C)O3)=O)CC=CC2)=O)CC(C)(C)C12CCC2 C(CC(C)(C)C(=O)NCC1(O)CCCOC1)NC(CC1(C)CCCCC1)=O C(=O)(C(=O)C(C)(C)C)NCC1N(C(c2nc(C)n(C)c2)=O)CCC1 C1(C(C)(C)C)(CNC(c2ccsn2)=O)CCN(C(=O)C=C2CCC2)C1 c1(C(=O)NC(C2CN(C(=O)C=CC3CCCO3)CCO2)C)ccc(S(C)(=O)=O)[nH]1 N1(C(C2OCCN(CC)C2)=O)CCCC12CCCN(C(=O)C1=C(C#N)CCC1)C2 CON1CCC(N(C)C(c2ccc(CNC(c3cn[nH]c3)=O)o2)=O)CC1 C(=O)(CCCCC(=O)N1CCC2(C1)CN(C(c1cnnc(C)c1)=O)C2)OC N1(C(c2c(C)noc2N)=O)CC2CCC1C(NC(=O)C(N1CCOCC1)C)C2 c1(C(=O)OC)cnc(=NCC2CCCCN(C(C3C(C)(C)C3(C)C)=O)C2)[nH]c1 C1(NC(CC(CC)(C)C)=O)CC2CCC(C1)N2C(C1C2CCC12)=O C1(C(=O)NCC(CC=C)NC(=O)Cc2ncoc2C)OCCCC1(C)C C(=O)(CC(F)(F)C(F)(F)F)N(CCCCNC(C1CC2(CCCC2)CO1)=O)C C1(NC(CSS(C)(=O)=O)=O)CC2COCC(C1)N2C(C1CCCC12CCC2)=O C1(C(=O)NC2(C3CN(C(c4n(C)ccc4)=O)C3)CC2)Cc2ccncc2C1 c1(C(N(CC(CN(C(CCCSC)=O)C)O)C)=O)cccc2c1OCC2C c1(OCCC)c(C)cc(C(C(=O)NC(C)C)N(CC(C(F)(F)F)OC)C)cc1C C1(CNC(CC(C=C)CC)=O)CC2(CO1)CN(C(c1ncc(C(F)(F)F)s1)=O)C2 C1(C#N)(C(N(CCN(C(C)C)C(c2coc(Cl)n2)=O)C)=O)CCCCC1 c1(C(=O)NCC(=C)CCNC(=O)CNS(N)(=O)=O)cccnc1N(C)C C1(OC)CC2CC1CN(C(C1CCN(C(=O)C3=CCCCO3)C(C)(C)C1)=O)C2 C1(CNC(c2scc(C)c2C)=O)CN(C(c2ccsc2C)=O)CCCO1 C1(NC(C2(C=C)CCC2)=O)CN(C(c2snc3ccccc23)=O)C2CCCCC12 C=CC(C)(C)CC(=O)N1CC2CC2(NC(=O)C(C)S(C)(=O)=O)C1 N1(C(C2CCC(C)C(C)C2)=O)CCC2CCC(C1)N2CCC(N1CCCCC1)=O c1(C(c2nnnn2CC2CC2)NC(CC=C)C)ccc(OC(F)F)c(Cl)c1 Cc1cc(C(N2C(CC(=O)NC3CCN(C)C(C)C3)C3CCCC23)=O)cc(C)c1 C(CC(=O)N(C)C(C)C(C(C)=O)CC)(C(F)F)NC(C(C)N)=O n1(C(COC)C)cc(C(N2CC(OC)CC2CNC(c2cnco2)=O)=O)c(C)n1 N(C(=NCCc1ncn(C)n1)NCC1CCC(CO)O1)C(c1ccccc1)C N1(C(c2ncn(CC)n2)=O)CCCC2(C1)CN(C(C1CC(C)CO1)=O)C2 Cc1cc(Cl)nn1-c1ccc(CNCCCN(CC(C)C)C)cc1 C1(c2n(CCCOC)nnn2)(NCCC2(C)COC2)CC2CC1CC2(C)OC N1(C(C=CC(CC)=CC)=O)CC2CCCC(NC(c3n[nH]cc3OC)=O)C2C1 c12ccnc(Cl)c1CNC(=O)N(C)CCCCSC2=O.C(C)(C)(C)OC.CO c1(C(=O)NC2C(CC)N(C(C3CC3OC(C)(C)C)=O)CC2)scc2c1OCCO2 CCCC(C)(O)C(=O)NC1COCCN(C(=O)C=C2CCC(C)C2)C1 C1(CC(=O)NC(COC)CCO)CCN(C(=O)C(C#N)C(C)C)C1(C)C c1(SC)ccc(N)cc1C(=O)NC1CCCC(NC(c2ccoc2)=O)C1 CC1(C)C2CCC(C2)C1(C)C(N1CC(NC(c2cn(C3CC3)cn2)=O)C1)=O c1(OC)cscc1C(=O)NCc1cc(C(=O)NCCC2CCC(C)O2)co1 C1(NC(c2ccc(Cl)cc2Cl)=O)CN(C(c2cc(O)cc(=O)o2)=O)C2(CCC2)C1 c1(OCC)cnc(C(=O)NCC2CN(C(c3ccc(CC)cc3)=O)C3CC23)cn1 C=C(C)CCC(=O)N1CCN(C(=O)CNC(=O)CC(C)NCC)CC1 c1(C2C(N3CC(c4nnc(-c5n(C)ccn5)o4)OCC3)C2)c[nH]c2ccccc12 C12(C(=O)NCCC3(O)CN(C(c4ccc(F)c(Cl)c4)=O)C3)CCCCC1C2(F)F c1(N2CCN(CCCOC)CC2)[nH]c(=NC2CCOC(C)(C)C2)nc2scnc12 N1(C(=O)C(c2ccccc2)Sc2nc[nH]n2)CCCC(c2ccon2)C1 N1(C(C(C=C)(C)O)=O)CCOCC2(COCCN2c2nc(-c3ccsc3)ns2)C1 c1(CNCc2ccc(C)nc2)cc(C)n(-c2ccccc2Oc2ccccc2)c1C C1(CC)CC(C)CN(C(=O)C(C)N(C)C(C2CCOC2C(C)C)=O)C1 N1(C(c2ccc(SC)s2)=O)CCN(C(=O)CC=C(C)C)CC1CC(F)F N1(C(C(C)=CC)=O)CC(CNC(=O)CCN2CCC(N(C)C)CC2)CC1C C(=O)(CCCN=[N+]=[N-])NC(C1COC1)=O.c12ccccc1NC(=O)C1C(C1)N2C N1(C(C(C)OCC(F)(F)F)=O)CC2(CCN2C(c2cncn2C)=O)C1 N1(C(c2c(OC)nsc2OC)=O)CC2(CCCC2NC(C2C3CCCCC23)=O)C1 CCC(C)(C)C(C)CC(=O)NCC(C1CC1)N(C(=O)CSc1ccc(F)cc1)C C(=O)(CS(=O)(=O)C(C)(C)C)NC1CN(C(CC(=C)C)=O)CC1CC1CC1 Cc1ccccc1CCC(N1CC(CNC(C2(c3cc[nH]n3)CC2)=O)CC1C)=O CCCC(C)CC(=O)NC1CCN(C(c2cc(C3CC3)on2)=O)CC1OC C(=O)(C(C)C(O)CCCC)NC(CC#C)C(=O)NCc1cc(C)nc(C)c1 C1(NC(C(N)=O)=O)CCC(NC(C2CC2NC(=O)OC(C)(C)C)=O)CC1 C12(C(N(C3CCOCC3)C)=O)CC(CO1)N(C(C1CC3CCCC3C1)=O)C2 N#Cc1ccc(C2CCCN(c3cc(-c4ccc(Br)cc4)nc(Cl)n3)C2)cc1 c1(C(=O)NC2CCC(NC(c3c(SCC)cccn3)=O)CC2)cnc(O)nc1O CC1CCCC1C(=O)NCC(C1CC1)N(C)C(c1cncn1C)=O CCC(C)(CNC(=O)COCC1CCCO1)NC(C1CC(F)(CO)C1)=O C1(c2cc(C)[nH]n2)CCN(C(=O)CC2(C)CC2(F)Cl)CC1 N1(C(C2(C=C)CCC2)=O)CCCC(C2CN(C(c3cc(C(N)=O)co3)=O)C2)C1 c1(N2CCC(OCC#N)CC2)nc(=NCc2cc(CO)co2)[nH]c2ccccc12 C(C)(C)(CCCNC(=O)CC1(O)CCCC1)NC(c1c(C)ocn1)=O C12(OC)CCC(CNC(=O)OC(C)(C)C)(CC1)C2.N12CCC(O)C(C1)C2 c1(NCCOc2c(OC)cccc2)c(O)cc(F)cc1F.C1(C)CNC(=O)N1 N1(C(c2c[nH]cc(Cl)c2=O)=O)CCCN(C(=O)C(O)Cn2cncn2)C(CO)C1 C1(CC=C)(C(=O)N(C)Cc2ccns2)CCCN1C(=O)CC1C(C)(C)C1(C)C N#Cc1ccc(C(=O)NC23CC(CNC(=O)COc4ccsn4)(C2)C3)s1 C(=O)(C1Cc2c(Cl)cccc21)N1CCN(C(c2cc(C)c(C(F)F)nc2)=O)CC1 C(=O)(C(F)CC(C)(C)C)N1CC(SC)C(C(N2CCC(OC(C)=O)CC2)=O)C1 N1(C(CCS(=O)(=O)NC)=O)CC2OCCN(C(c3ccc(=O)oc3)=O)C2C1 C12(C(=O)NCCNC(c3cc(Cl)c(O)c(Cl)c3)=O)CCCN(CC1)S2(=O)=O N1(C(c2c(C)noc2)C2CC2)CC2C3CCC(C2C1)N(C(=O)COCC(F)(F)F)C3 CC(C)CCCC(C)N=c1ccc(S(=O)(=O)NC2CC(C)(C)OC2(C)C)c[nH]1 c1(C(N2CCC(NC(C3(CC)CC3(F)F)=O)C2)=O)cc(COC)nn1CC1CC1 N1(C(c2c(C(N)=O)coc2)=O)C2CCC1CN(C(c1ccc(OCF)cc1)=O)C2 N#CC1CN(C(=O)CCCCCl)CC1NC(=O)Nc1ccc(Cl)cc1 C(=O)(CCC(CC)NC(=O)CCCC1CC1C)N(CCCN(C)C)CCC C1(C(=O)NCC(C2CC2)NC(c2c(C)nn(C3CC3)c2)=O)CC2(CCC2)CO1 N(C(=NCC1CCOC1)NC(C)C)C(CC)CC.C(=O)(C)OC CC(C)(C(=O)NCC1CN(C(=O)CCNC(C2CCCCC2)=O)C1)c1cncs1 N1(C(c2nnc(C(C)C)s2)=O)CCC(C2CCN(C(=O)C(C)C(C)O)CC2)C1 Cc1cc(C(N2CCC(F)CC2C(=O)NCc2ncsn2)=O)cc(C)c1 C1(C(=O)OC)CCC(C(N2CCCC2CN(C)C(c2nc(Cl)cs2)=O)=O)C1 CC(C)(C)C1=NOC(C)(C(N2CC(NC(=O)CN3CC=CC3)C(C)(C)C2)=O)C1 c1(OC)cccc(N2CCCC(NC(=NCc3ncn(C)n3)NC3CC3)C2)c1 CC(C)C(C)C(CNC(=O)CC1(CO)CCOCC1)NC(=O)CN1CCCC1 Cc1cccc(C(C)C)c1C(=O)NC1CN(C(C2CC=CCO2)=O)CC1C(F)F C1(CNC(C(CCOC)(C)C)=O)CC2(CCN(C(c3coc(CO)c3)=O)C2)CO1 c1(OC)cc(C(=O)NC2CC2C(=O)Nc2ccc(O)cc2Cl)ccc1C Cc1cc(C)c(CC(=O)NCCNC(=O)C2=COCC2)c(C)c1 c1(CN(C(=O)C(=O)NCC(F)F)C)cccc(CNC(=O)CC2CCC(=O)N2)c1 N1(C(CCCC#CC)=O)CC(C(=O)NCCc2cc(C)[nH]n2)CC(C)(C)C1 CCC(CCOC)C(=O)NC1CCN(C(=O)C(F)(F)C2CC2)CC1O C(=O)(CCCC(=O)N1CCC(F)(C(=O)NC(C)(C)CC(F)CO)C1)OCC C1(C(N(CCN(C(CCC#C)=O)C)C)=O)CC(C)N(C)C1 c1(C(=O)NCC2N(C(c3ccc(Cl)s3)=O)CCCC2)cc(F)cc([N+](=O)[O-])c1 Cc1noc(C(F)(F)F)c1C(=O)N(C1CCN(C2CC2)C1)C c1(CC(=O)NCC2CCCC(NC(C3C4CCCOC34)=O)C2)ccc(F)c(Cl)c1 C#CCC(CC(=O)N1CCCC(C(C)(C)C)C1)NC(=O)C(C)(C)CCC N1(C(C2CCNC3(CCC3)C2)=O)CCN(Cc2ccccc2)C2CCCC12 C(=O)(C1Cc2ccccc21)N1CCC(OCC2(CC(=O)NCCOC)CC2)C1 c1(C(C)(C)C)ncc(C=CC(=O)NCC2CC2NC(=O)Cn2cc(CO)nn2)s1 CCCCC(C(=O)NCCCCC(C)(C)NC(C1CC(OC)C1)=O)C(C)C Cc1ccc(O)c(C(=O)NCC(n2cc(CN3CCN(C)CC3)nn2)C)n1 C(=O)(C1=C(C)N(C)c2ncnn2C1C)N1CCC(NC(CCOC)=O)C1C(C)C c1(C(=O)NCC2C(C(=O)NCC(=O)NCCC)CCC2)cc(C)ncc1C c1(-c2ccc(C(=O)NCC3(C)OCCO3)nc2)ccc2c(c1)CCCO2 N1(C(C(C)NC(=O)NC(c2ccco2)=O)=O)CCC(NC(=O)Cc2ccsn2)C1 N1(C(C)=O)CC(O)(CC(C2CC2CC(C)C)=O)C1.c12cn(nn1)CCNC2=O CCC(CC)(CO)C(=O)N1CCN(C(C2C(C(F)(F)F)C2[N+](=O)[O-])=O)CC(O)C1 C1(NC(CCCC)=O)CC2(CCC(CNC(=O)CCC(F)F)OC2)C1 c1(C(=O)NCC2(C)CCN(C(c3cnc(C)s3)=O)C2)ccc2nc[nH]c2c1 C1(NC(Cc2n(C)ccn2)=O)COC2C(NC(=O)CC3CCC(=O)CC3)COC12 C1(C(=O)NC(CCSC)C(=O)NC(C)C)CCCCCCC1.C12(CC1)C(=O)N2 Cc1cc(C(N2CCC(NC(c3ccc(=O)n(C(C)C)c3)=O)C2)=O)c(O)c(C)n1 c1(C(N(CCC)CCNC(=O)C(F)CC2CC2)=O)cncc(C(C)=O)c1 C1(C)(CNCc2cc(C3(C)CC3)on2)CCCN(C(=O)C(O)C2CC2)C1 C1(C(=O)NCC2CC(NC(c3sccc3SC(F)F)=O)C2)CCCC2CCCN12 C1(C)(C(=O)NC(CC)CNC(c2ncoc2-c2ccon2)=O)COC(=O)OC1 c1(C(=O)NC2(C)CCN(C(c3cc(C(C)=O)oc3)=O)C2)c2ccccc2nn1C c1(C(N2C(C)CC(CNC(=O)C(C)(C)C3CC3)C2)=O)ccc2nc[nH]c2c1 c1(CN(C(=O)C(O)C2CC2)C)ccc(CNC(c2ncoc2C2CC2)=O)cc1 C1(C)(NC(CCOC)=O)CC(NC(c2ccc(CCCCCC)s2)=O)C1 c1(OC)cc([N+](=O)[O-])c(NC(c2sccc2NC(c2ccsc2Cl)=O)=O)cc1C N1(C(C2C=CCC2)=O)CCCC(N=c2[nH]c3ccc(O)cc3s2)CC1 N1(C(Cc2ccc(C)s2)=O)CCC(CO)(NC(=O)CC2CSCCS2)C1 c1(C(=O)ON)cccc2[nH]c(-c3cccs3)nc12.CC12CN(C1)C2 c1(C(N2CC(CNC(Cc3ccn(C)n3)=O)CC2(C)C)=O)cc(Cl)c(F)c(Cl)c1 c1(CC)cccc(CN(C(=O)C(N)c2cscn2)C2CC2)c1 C1(CC(=O)Nc2nn[nH]n2)CCCN(C(=O)CCc2nc(Br)cs2)C1 CC(C)C(C)(C)C(=O)NCCC1(C)CCN(C(=O)CCC(=O)N(C)C)C1 CC1(C)CCN(C(C2CSC2)=O)CC1C(=O)NCCN=[N+]=[N-] CCCCCCC(O)CCC(=O)NC1CN(C(C2CC2C(=O)OC)=O)CCC1C C1(C(N(CCCOCCNC(C(CC)SC)=O)C)=O)Cc2cccc(OC)c2O1 C#CCC(O)C(=O)N(C1CN(C(=O)Cc2ccc(Cl)cc2)CC1O)C n1(CC(N2CCC(NC(C=COCC)=O)C(C)C2)=O)cnc2c1CCCC2 N1(C(CC2C(C)CCO2)=O)CC2CCC(C1)N2C(=O)CCN1CCCS1(=O)=O N1(C(CSCCC(C)C)=O)CC2(CNC(c3nocc3Cl)=O)CCC1CC2 C1(C)(CNC(c2cn(C)nc2O)=O)CN(C(c2c[nH]c(=N)o2)=O)C(C)(C)C1 c1(C(N2C(CNC(C(c3cn(C)nc3)O)=O)CC2)=O)cccc(=O)n1O Cc1cc(Cl)c(C(=O)NC2CC(C)N(C(=O)C=Cc3ccccn3)C2)cc1C C(=O)(C1CCCc2cn(C(C)C)nc21)NC1(CO)CN(C(C2C(COC)C2)=O)C1 n1(C(C)C)nc(C2CC2)cc1C(=O)NCC1CC1NC(=O)CCCn1cccc1 Cc1cc(NC(C2CCN(C(=O)C3=CCC(C)CC3)C2)C)n2ncc(C)c2n1 c1(CNC(C(C)n2ccnc2)=O)ccc(C(=O)NC2CCC(O)CC2)cc1 c1(C(=O)NCC2CN(C(C(C)(C)C3CCCC3)=O)CC2O)cc(Cl)nnc1O N1(C(C(COC)NC(=O)CCCN(C)C)=O)CCCC(N=[N+]=[N-])CC1 c1(CN2C(C(=O)NCc3n[nH]cc3Br)CC(F)C2)cn2cccnc2n1 CC1(C)CCCN(C(=O)COc2ccc(F)cn2)C1CNC(C1(C)CCCO1)=O C(=O)(C(C)C(O)C(C)C)N1CC(SC)C(NC(=O)CCc2nnc(C(C)C)o2)C1 C(=O)(C(C(C)(C)C)NC(=O)Cc1ccn(CC)n1)N(CC(=O)OCC)C CC1CN(C(C2(NC(=O)C3=CCCCC3C)CCOCC2)=O)Cc2c[nH]nc21 N1(C(CC)=O)CCC2CCCN(C(c3cnn4cc(OC)ccc34)=O)C2C1 CN1Cc2ccc(C(N3CCN(c4cncs4)CC3)C(=O)NC3CC3)cc2C1=O c1(NCc2cnnc(C)c2C)cc(Br)ccc1S(=O)(=O)NCC1CCOC(C)C1 C1(C(N(CC(CNC(CCC(=O)NCCC)=O)C)C)=O)CC(=O)CC(=O)C1 Cn1[nH]c(=NC(=O)C2CCC(c3ncc[nH]3)CC2)cc1C1CCOCC1 C1(CC)CCC(C(=O)NCC2CN(C3(CNC(=O)C(CC)SC)CC3)C2)CC1 C1(NC(C2CC3CC3C2)=O)CC(N=c2[nH]nc(C(F)(F)C(F)(F)F)o2)C12CCC2 c1(C(N2C(CC(N3CCCC(CC)CC3)=O)CCC2)=O)ccc2c(c1)CCC2 c1(COC(C2N(CC)CCC2)=O)ccc(CCNC(=O)OC(C)(C)C)c(C)c1 C12(NC(CC3CC(=O)C3)=O)CCCC(NC(=O)CC(O)c3ccccc3)(C1)C2 CC1CN(C(=O)CCC(=O)N(C)C)CCC1N(C(=O)CCc1ncc[nH]1)C C1(C(=O)NC(C)CCN(C(=O)C(C2CC2)C2CC2)C)(OC)CCCCC1 C1(C(=O)NCCC(CNC(c2nn(C)c(F)c2)=O)(C)C)CC(C)(C)OC1(C)C C1(CNC(C2C(C)OCC2)=O)CN(C(c2ccnc(S)c2)=O)CC12CCOCC2 Cc1c(C(=O)N(c2ncc(C#N)s2)C2CC3(CNC3)C2)cc(F)cc1[N+](=O)[O-] Cc1cccnc1C=CC(=O)NCC1(CN(C(=O)CC2CC2C)C)CC1 C1(C)(CNC(C(C)OCCC=C)=O)CCCN1C(c1ccc(CC)o1)=O CCC(CC(F)(F)F)C(=O)N1CCC(NC(=O)CCC=CC(C)C)C(CO)C1 C1(O)(CN(C(CSCC#C)=O)C)CCCN(C(c2cc(C(=O)OC)nn2C)=O)C1 C1(NC(c2cnc(O)o2)=O)CC2C(NC(C3CCCSC3)=O)C2C1 C1(NC(CCOC(CC(C)C)C)=O)CN(C(c2cc(C3CC3)ns2)=O)CC1(C)C c1(C(=O)NC2CCCN(C(C34CC(OC)C3C4)=O)C2)ccc(N)c(Cl)n1 C1(C(=O)NC(Cn2ncc(C)c2)C)CCC(C)CN1C(=O)C(O)CN(C)C c1(C(=O)NC(CC)CN(C(=O)C2=CC(C)(CC)C2)C)nnn2c1CSCC2 N(C1CC(C)n2ccnc21)c1ccc(N(CC)CC)cc1 C1(C(N2CCC(CNC(C(CCC)N(C)C)=O)C2(C)C)=O)CCc2nnnn2C1 c1(C(=O)NC(CNC(c2c(C)cns2)=O)CC(C)C)ccc2c(c1)C(C)(C)CN2 CC(C(C)(C)C(=O)NCC1CC1(C)C)NC(c1ccc(O)cc1F)=O N1(C(C(C(CC)C)OC)=O)CCC2(CC(NC(C3(S(C)(=O)=O)CC3)=O)C2)C1 C(=O)(CC(C)C(F)F)NC(C1CN(C(C(N2CCC(C)CC2)=O)=O)C1)C c1(C(=O)NC(C)CCCCNC(=O)CN(C)C(N)=O)ccnc(O)c1Br c1(C(N2CC(O)(CNC(C(C)NC(C3CCC3)=O)=O)C2)=O)cc2c(s1)COCC2 N1(C(CC2CC(C(C)C)OCC2)=O)CC2(CNC(C3CC(O)C3)=O)CCC1CC2 n1(CCF)nc(-c2ccc(Cl)cc2)nc1-c1cccnn1 C1(C(=O)NCCc2ccc(C)c(C)c2)CC12CCN(Cc1ccc(Br)[nH]1)CC2 c1(C(=O)NCC(CC=C)NC(c2c(C)[nH]c(C)c2C)=O)csc(=NC2CC2)[nH]1 CC(C)CCC(C(=O)N1CC2(CCCO2)C1)NC(C1CC2CCCC2C1)=O C(=O)(C1=CCCCC1)N(C1CCN(C(c2cnn[nH]2)=O)CC1)C C1(CNC(C(C#C)(C)C)=O)CCC2(CCN(C(=O)CN(C)C(C)C)CC2)CO1 c1(C(=O)NC(CCC)C(=O)N(C2CCOC2)C2CC2)cc2n(n1)CCO2 C(=O)(C(C#N)C(C)(C)C)NCC(CC(=O)N1CC(OC(CC)=O)C1)O C(=O)(C1=C(Cl)CCOC1)NCc1c(C(=O)NCC2CCCC(C)(C)C2)[nH]cc1 C(CC(C(C)(C)C)NC(c1cnn(C)c1Cl)=O)N(C(c1c(C)cc(F)s1)=O)C S(=O)(=O)(c1ccc(N(C)CC2CC(F)C2)cc1Cl)NC(CCC)CCO C1(NC(=O)NC2CCN(C(=O)C(=O)OCCCOCC3CC3)C2)CC12CCOC2 c1(C(=O)NC(C)CN(C)C(c2cnns2)=O)cn2cccnc2n1 CC(C)CCCC(C)CNC(=O)CCn1cc(CS(C)(=O)=O)nn1 c1(OCC)cccc2cc(-c3cn(CCNC(C4CC(CC)C4)=O)nn3)cnc12 CC(F)(CNC(c1ccnn1CC1CC1)=O)CNC(C1(C)CCOC1)=O N(C(=NCC1CCCC(C)(C)C1)N1CC(O)C2(CC2)C1)CC(C)C c1(OC)cc(CNCCC2CC(F)(F)CN2)cc(C)c1 Cc1cccc(OCC(=O)N(CCNC(=O)C(O)C2CCCC2)CCOC#N)c1C CC(CCNC(=O)CCCCN1CCOCC1)CCNC(C1CN(C)CCO1)=O CC(C)CC(CNC(c1cnc(C(C)C)o1)=O)NC(C12CCC(CC1)C2)=O N1(C(c2cc(C(C)=O)on2)=O)CCC(CN(C)C(C2(C)CCSCC2)=O)CC1 CC(C)C(O)C(=O)NCC1CCN(C(=O)CCS(C)=O)C1 N=c1nc[nH]n1CC(=O)NC1CCN(C(C2CCC(c3cc[nH]n3)O2)=O)C1 C1(CC=C)(C(=O)NCCC2COCCO2)CCN(C(c2cc(C)c[nH]2)=O)C1 C1(OC)CCN(C(=O)CNC(C2CN(C(=O)C(C)(C)C)C2)=O)C1(C)C c1(C(N2C(C)CCN(C(c3ncccn3)=O)CC2)=O)noc2c(F)cccc12 C1(NC(C2(CC=C)CCOCC2)=O)CC2CCC1C(NC(c1ccsn1)=O)C2 N1(C(c2cc(COC)sc2)=O)CCC(CCCNC(c2cccc(=O)o2)=O)CC1 C(=O)(C(CO)C(F)(F)F)NCC(CC=C)C(=O)NCC1(CO)CC(C)C1 C1(C(=O)NC(C(=O)N(CC(C(C)C)OC)C)Cc2cc[nH]n2)CCCC(=O)C1 N1(C(CN(C)CCO)=O)CCC(C(F)(F)F)CC1CNC(=O)CC1OCCCO1 C1(CCOC)(NC(c2cccc(CO)n2)=O)CCN(C(C2CC2C#N)=O)C1 C1(CC#C)(C(=O)NC(CNC(=O)C(c2cccn2C)=O)(CC)CC)CCOCC1 C=C(CNC(c1sccc1F)=O)CCNC(C1(O)CC(c2ccccc2)C1)=O c1(OC(COCC)=O)ccc(OC2CC(C)N(Cc3ccccc3)C2)cc1C C1(NC(Cc2c(C)ocn2)=O)CCOC12CCN(C(=O)C#CC1(C)COC1)CC2 C1(CNC(c2c(C)nn(C)c2)=O)CN(C(=O)CCC2CC2C)CCN1C CC1C2C(CCN2C(C2CC(F)C2)=O)CN1C(=O)C1=NNC(=O)C1 C(=O)(C(CCC)C(=O)OC)NCc1cc(C(=O)NC2(C=C)CCOCC2)sc1 c1(SC)cccnc1C(N1CCC(C)(NC(=O)CC2CCC(=O)N2)C1)=O C1(CCC)(NC(c2occ(C)c2C)=O)CCN(C(=O)CC2COCC(C)O2)CC1 c1(C(=O)NCC2C(CNC(CCCC(C)(C)C)=O)C2)cccc2[nH]nc(O)c12 S(=O)(=O)(c1cc(C(=O)O)cc2c1OCC2)NC(c1cc(-c2n(C)ncc2)[nH]n1)=O C(=O)(C#CC1CCCC1)N(C)CC1CCCC(NC(c2cc(F)cc(Cl)c2)=O)C1 N1(C(C(C)O)=O)CCC2(C1)CN(C(c1c(F)cc(O)cc1F)=O)CC(C)O2 C1(NC(C2CCN(C(CC)=O)C2)=O)CC(C)CN(C(c2cnc(C3CC3)s2)=O)C1 CC1CN(C(=O)COC2CCCCCC2C)CCC1C(=O)NC1CC=CC1 C1(OC)(CNC(C2CC3CCC3C2)=O)CCN(C(c2cnn(C(C)C)c2)=O)CC1 c1(C(=O)NC(C(C)C)CCO)c(F)c(F)cc(F)c1F c1(C(=O)NC2CCC3(CN(C(CCN(C)C)=O)C3)C2)cc2cc(Br)ccn2n1 N1(C(CN(CC(C)(C)C)C)=O)CC2(CCCC2CC(N2CCCC(F)C2)=O)C1 C1(NC(COC(CC)C)=O)CC2COCC(C1)C2NC(C1CC(C)(C)C1)=O N1(CCNC(C2C(CNC(c3cc(CC)on3)=O)CCC2)=O)CCCOCC1 c1ccc(-n2cc(CCNCCCn3ccnc3)nn2)cc1 N1(C(C2(SC)CCC2)=O)CC2(NC(c3ccnc(C4CC4)c3)=O)CCC1CC2 O=Cc1sc(CN2CCCC(C(N3CC(O)C(F)C3)=O)C2)c(Br)c1Br c1(NCCN2CCN(C(=O)CCN3CCCCC3)CC2)cc(F)cc(F)c1Br.OS N1(C(C(CCC)(C)O)=O)CC2(CC(C(=O)NC(C3CCOCC3)CC)CO2)C1 c1(C(=O)NC(CCN(C(CC(CC)C2CCC2)=O)C)C)cccc2oc(C)nc12 Cc1oc2ncnc(O)c2c1C(=O)N(CC(C)(C)CNC(C1CCC(C)O1)=O)C N1(C(C(=C)F)=O)CCC2(CC(C(=O)Nc3cc(O)ccc3Br)=NO2)C1 C1(C(N(C)CC2C(C)C2)=O)CC(NC(C2CN(C)C2)=O)C(O)C1 C(=O)(C(CC(C)(C)C)NC(=O)C(C)CC(=O)OC)NCC(=C)Br C1(NC(C2(CCCC)CC2)=O)CCC2(CCCN2C(c2cc(C)on2)=O)CC1 C(=O)(C#CC1CN(C(=O)OC)C1)N1CCC(C)(CNC(C(C(C)(C)C)OC)=O)C1 C(=O)(CC(C)C(C)(C)NC(C1C=CCCC1)=O)NC1C2(CC(OCC)C2)C1 Cc1cncc(CNC(=O)C(C)N(C(C2(C)CCCOC2)=O)C2CC2)c1 Cc1cn2nnc(C(=O)NCC3C4CN(C(c5conc5C)=O)CC34)c2c(O)n1 C=CC1CCCN1C(c1csc(C2CC2)n1)C(=O)NCCCF C1(N(C(=O)Cc2csnn2)C)CCCC(NC(=O)CSc2ccnn2C)C1 C1(NC(C2(NC(c3[nH]c(=N)sc3)=O)CCCCC2)=O)CC2C(O)C(O)CC12 C(=O)(CC1=CCN(C)CC1)NC(CC(C)NC(c1ccc(-c2cccs2)[nH]1)=O)C Cc1cc(C)c(C(=O)NCCCCNC(C2CCCCN2S(C)(=O)=O)=O)[nH]1 C(=O)(C1COc2ccc(F)cc21)N1CC2(CCN(C(C(C)OCC)=O)C2)C1 c1(C(=O)NC2CCCN(C(CC3CC(CC)C3)=O)CC2)cc(N)c(N)cc1F C1(OC)(CNC(=O)Cc2cc(-c3ccccc3)on2)CC(C)C1 c1(C(=O)NCC23CC(NC(CCSC)=O)(C2)C3)sc(C(C)(C)C)nc1C C(=O)(CCCC(=O)NOC(C)(C)C)N1CC(NC(C(C)SC)=O)C(CO)CC1 N1(C(CC)=O)CC(CO)C2(C1)CN(C(c1c(N)cccc1Cl)=O)C2 Cc1ccc2occ(CC(=O)NC3CC4CN(C(C5CCOC5)=O)CC34)c2c1 c1(C(=O)NC(C(=O)N(C2(COC)CC2)C)CC2CC2)cccc2c[nH]nc12 C=CCCC(CC(C)C)C(=O)N1CCC(NC(=O)CCSC(F)(F)F)C12CCC2 C1(C(=O)NCCOC(CC)CC)CCC(C)(C)N(C(=O)CC2CC3(CC3)CO2)C1 c1(C(N(CC(C)NC(C23CC(F)(C2)C3)=O)CC)=O)cn(C)nc1Br c1(C(=O)NC(C)CCNC(C2CC2C(F)(F)F)=O)cc(-c2ccccc2)on1 c1(CC)conc1C(=O)NCC(C)(C1CCC1)NC(=O)C(C)Cc1ccnn1C c1(CCC(C)O)cn(CC(=O)N(C2CCN(C(C3CC3F)=O)C2)CCO)nn1 c1(CNC(c2ncccc2-c2ccc(CO)nc2)=O)ncc(C(F)(F)F)cc1F C1(N=c2nc3[nH][nH]cc-3c(O)n2)(COC)C2CCCC(C2)N1C(=O)OC(C)(C)C Fc1ccc(F)c(CNC(c2nnnn2C2CCCC2)c2csnn2)c1 N1(C(C(C=C)O)=O)CCN(C(c2ccc(Cl)c(CC)c2)=O)CC1CO Cn1ccc2ccnc(C(=O)NC3(CCCNC(C4(O)CCCCC4)=O)CC3)c12 CC1CCN(C(=O)C(C2CCC2)C2CCC2)CC1CNC(c1ccccc1O)=O c1(CCC)ncoc1C(=O)NC(C(=O)NCCN(CC(F)F)C)C1CC1 c1(NC(=O)NCCS(C)(=O)=O)ccc(Cl)c(NC(C2(F)CCNCC2)=O)c1 C1(NC(Cc2c(C)cccn2)=O)CCCC12CN(C(=O)C(C)Cn1cccn1)C2 CCCC(C(=O)NC(C)(CNC(=O)Cn1ncc(Br)c1C)CC)NC(N)=O Cc1cc(C(=O)N(CC(=O)NC2(c3ccncc3)CC2)C(C)C)cc(O)c1 Cn1nccc1C(C(=O)NCc1cc(O)ns1)NC(=O)CC12CCCC1C2 N1(C(c2[nH]nnc2C)C(=O)NCC(=C)C)C2CCC1CC1(C2)N=N1 Cc1cc(C(N2CCC(CNC(C34C=CC(CC3)C4)=O)CC2)=O)cc(=O)n1C Nc1ccc(S(=O)(=O)N2CC(CC3CCCCCC3)C2)nc1 c1(C(N2CCN(CCN(C(c3occ(C)c3)=O)C)CC2)=O)cnn2ccn(C)c12 c1(OC)cn(C)c(C(=O)NCC2CCC(NC(C34CCC3C4)=O)C2)cc1=O c1(C(=O)NCC2(CCNC(C3C(=C)C3)=O)CC2)ccc(N=[N+]=[N-])cn1 C1(C(=O)NCCC(=O)NCC#C)CCC(NC(=O)CC(C)F)C1 N1(C(c2n[nH]c(C)c2Cl)=O)CCC(C(N2CCC(C)(F)C2)=O)C1(C)C N1(C(c2ccc(NC)cn2)=O)CC2(CNC(=O)C(F)(F)C(F)F)CC1CO2 c1(C(=O)NCC2(NC(=O)CC3CCC(F)(F)C3)CC2)cccc2c1CCS2(=O)=O c1(C2C(C)C2)ccc(-c2nc(C3CC34CC4)nn2-c2nccn2C)cc1 C=CC1OCCC1C(N1CCN(C(C)CNC(=O)C(O)C2CC2)CC1)=O C1(c2ccccc2)(CC)CN(CCC(=O)NC2COC(C)(C)C2)CCO1 N1(C(C(C)CNC(=O)C(C)(C)N=[N+]=[N-])=O)CCC2(CNC(=O)C2)C1 C1(CNC(CCC(=O)NCC)=O)CN(C(C2C(C)C2C)=O)CCC12CCC2 N1(C(C2C(NC(CC(C)(C)C)=O)CCO2)=O)CCOCC(O)C1 C(=O)(CCS(N)(=O)=O)NC1CC(CC(=O)NCC(=O)OCCCC)C1 C(=O)(NN1CCCC1C(=O)NC1CCOC12CCCC2)c1cc(C)[nH]c1C C1(C(=O)NC(CC2CCN(C(CC(CC)OC)=O)CC2)C)CC(S(C)(=O)=O)C1 S(=O)(=O)(c1cnc(N2CCCC(CO)C2)cc1C)NC(CC)C(C)C c1(C(=O)NC2C(C)(NC(C(C3CC3)OCC)=O)CCC2)nc(C)ccc1C c1(CNC(C(=O)NC(C)CN(C)Cc2ccccc2)=O)ccc(F)c(Cl)c1F C#CCC(O)C(=O)N1CC(O)(CNC(=O)C(C)(C)SC)C1 N1(C(CCC2CCC(C)O2)=O)CCC(CNC(c2cccnn2)=O)C12CC2 C(C1(C)CCOCC1)=CC(=O)NC(C1CCCN(C(=O)Cc2ccc(Cl)s2)C1)C CC1OCCCC1C(=O)NC12CC(C1)N(C(=O)C(F)=C1CCCC1)C2 C1(C(=O)NCCCC(CCC)NC(=O)CCCCCC#N)CCn2nncc2C1 CC(C)(CF)C(=O)NCC1(C(C)(C)C)CCN(C(=O)CCCNC(=O)OC)C1 C(C#Cc1cnn(C)c1)NC(c1c(CNC(CCCCC#C)=O)cco1)=O C1(NC(c2nncc(CCC)c2)=O)CCN(C(c2cc(C(=O)OC)sn2)=O)C(C)C1 c1(CC(=O)NCCNC(=O)OC)cc(C2CC2)no1 C(=O)(C1(C)CCc2ccccc21)N1CCCC(COC)(NC(=O)CC(C)C)C1 N1(C(c2cnc(C)nc2C)=O)CCN(C(c2[nH]ncc2C#N)=O)CCC1C C1(CCNC(c2c(C)n(C)nc2)=O)CCCN(C(=O)CC(C)C(C)C)CC1 c1(CCC(=O)NCC2(OC)CN(C(C3C(CC)CCO3)=O)C2)cccc(F)c1F c1(N2C(C)CC(CNC(C(c3ccc(Cl)s3)C)=O)C2)ncnc(Cl)c1F C(C)(CCC(=O)N1CC(O)CC1CC(N1CCC(c2ncco2)C1)=O)OCC CCCC(O)C(CO)NC(c1cn(CCNC(c2cc(O)ncc2F)=O)nn1)=O C(CN(C)C)(C(=O)N(C1CCN(C(C)=O)C1)C)NC(C(C)=C1CCCC1)=O Cc1cc(F)cnc1C(N1CCN(C(C2C(C)C2C)=O)CC1c1ncc[nH]1)=O c1(CNC(C(C)OCC)=O)ccc(CN(C)C(c2ccc(CC)cc2)=O)cc1 CC(C)C(C)C(=O)NCC(C1CCCC1)NC(C1(C)CC(F)C1)=O C(=O)(C1CCc2ccc(Cl)nc21)NCCC(C)N(C(=O)C=CC(F)(F)F)C c1(C(N(C2CN(C(C(CC=C)CC)=O)CC2O)C)=O)cc2c(C)c(F)ccc2[nH]1 C1(n2cc(CCC(=O)OC)nn2)CC2CCC1(NC(c1cc(C(C)C)sn1)=O)C2 C1(C(=O)NC2(CSC)CC2)CCC1NC(=O)CCn1ccnc1 C1(N=[N+]=[N-])(C(=O)NCC(C(C)(C)O)F)CCN(C(=O)CCC2CC2(F)F)C1 Cc1c(F)ccc(CN2CC(C(=O)Nc3c(Br)cc(Br)cc3Br)CC(F)C2)c1Cl c1(N2CCC(OCCNC(=O)CC3(O)CCOCC3)C2)ncnc2cc(Br)sc12 Nc1ccc(C(N2CCN(C(C3(F)CCCCC3)=O)C(CF)C2)=O)cc1F c1(CC)cccc(C(N2CC(NC(C3(C(F)(F)F)CC3)=O)C3CC23)=O)c1O C(CC(C(=O)N(C(C)C(=O)NOCc1cccnc1)C1CC1)OC)OC n1(CC=C)nnnc1C(CCCOC)NC(=O)OC(C)(C)C C1(N(C(CC2(OC)CCC2)=O)C)CCCN(C(C2(O)CCC2)=O)CC1 c1(C(=O)NCCC(C(C)C)NC(C2CCCCC2)=O)cc(F)cc2cc[nH]c12 CCC(C(=O)OC)C(=O)NCC1(OC)CCN(C(=O)Cc2cnoc2)C1 CC1(C)C(NC(=O)CNc2ccccn2)CC1CNC(=O)C=Cc1cnccn1 c1(C(=O)NCC(C)N(C(=O)C=Cc2ccco2)C)ccc2c(c1)NC(=O)CS2 C1(C(=O)NC(C=CC(=O)N(CC#C)C(C)C)C)C(C(C)=O)C1(C)C N1(C(C2(C)CC=CCC2)=O)CCC(NC(C2CCC=CO2)=O)C(CO)CC1 C(CC(C)C)(C(=O)NCCCc1ccnn1C)N(C(C(=O)NCC)=O)C C1(C(N(C(C)C)C2CC2)=O)CC2CC1CC2NC(c1ccc(C(N)=O)[nH]1)=O O=C(C1=CCSC1)NC1CCCC1NC(c1c[nH]nc1-c1ccsc1)=O C(c1ccc(F)c(F)c1)=CC(N1CC(CCO)(CNC(CCC(=O)NC)=O)C1)=O c1(OCC(N2CCC(CCNC(c3cnc[nH]3)=O)CC2)=O)ccc(Cl)cc1Cl C1(NC(c2ccn(C)n2)=O)CN(C(C2CC23CCOCC3)=O)CC1S(C)(=O)=O N1(C(CC(CC)C)=O)CCN(c2nc(C(C)(C)C)nc(=N)[nH]2)CC(O)C1 C(N=c1[nH]ccnc1F)C1N(C(=O)C=Cc2cc[nH]n2)CCC1 c1(C(N)=O)cc(N2CCCC2CCCNC(c2ccc[nH]2)=O)nc(Cl)n1 CC(C)CCCC(=O)NCC1CCN(C(=O)CC2(O)CCN(C)CC2)CC1 N1(C(C2(O)CCSCC2)=O)CCCC2(CCN(C(C3(C(F)(F)F)CC3)=O)C2)C1 c1(OC)cccc(C(N2CC(C)C2C(N2CCC(C)CC2)=O)=O)c1 CC(C)CC(CC(=O)NC1CCCC1C#N)NC(c1cc(C#N)cn1C)=O N1(C(CCCN(C(CC(C)(C)OC)=O)C)=O)CCC2CCC(C1)S2 C1(C)(OC)CC(NC(C2CCCN(C(=O)C3=CCSC3)CC2)=O)C1(C)C CC1CCc2[nH]c(C(=O)NC3CCC3NC(C3SCCCS3)=O)cc2C1 c1(COC(C(C)Oc2c(C)nn(C)c2C)=O)nn(C)c2c1COCC2 CC1(C(c2nnnn2C2CCOCC2)NCCC#CCO)CCCCC1 C1(C)(CNC(CCc2onc(C(C)OCC)n2)=O)CCCN(C(=O)CC2CC2)C1 N1(C(C=CCC)=O)CCN(C(=O)C(C)(C)c2cnc[nH]2)CC1CF c1(OCC)cnc2c(CN3CCCC(O)CC3)cccn12 C1(O)(CCNC(C2CC3C=CC2C3)=O)CCCN(C(C2CCOCC2)=O)C1 N1(C(C2CCC(CC)C2)=O)CC(F)CC1C(N1CCCC(Br)C1)=O c1(C(=O)NCCN(CCC)C(c2n[nH]c(C)n2)=O)cn(C)nc1C1CCCO1 CCCCCCC(=O)N1CCC(CCOC)(NC(C2COCCO2)=O)C1 O=C1OC2CCN(C(c3c[nH]c(-c4ccncc4)n3)=O)CC2O1 C(=O)(C(O)CC(C)(C)C)NC(C)CN(C)C(c1nocc1-c1ccccc1F)=O N1(C(C2Cc3n(cc(C)n3)C2)=O)CCCC12CCN(C(=O)C(C)O)C2 c1(C(=O)NC2C(NC(C(=C(C)C3CC3)F)=O)CCOC2)cc(N)c(F)cc1C C1(CNC(C2CC2C2CCC2)=O)CN(C(=O)C=CCO)C2(CCOCC2)C1 N1(C(c2ccnc(C3CC3)c2)=O)CC2(C1)CN(C(=O)COC1CCCC1)C2 N1(C(CC2(C#N)CC2)=O)CCC(OCCNC(=O)CSc2cccc(Cl)c2)CC1 c1(N2CCC(O)(CC(N3CC4CCCC4C3)=O)CC2)ncnc2cc(I)sc12 c1(CN(S(=O)(=O)CC(F)(F)C2CCOCC2)C)ccn2ccnc2c1 C1(NC(C2C(C(=O)OC)C2)=O)CCN(c2cc(C)nc(C)n2)CC1C C(=O)(CS(=O)c1ccc(Cl)cc1)NCCC1CN(C(C2C(C)C2)=O)CC1C NS(=O)(=O)CC(=O)NC1CCC1CNC(C1(CC(F)F)CCOCC1)=O Cc1ccc(C(=O)NCCC(=O)NC2CCN(C(c3cc(Cl)ns3)=O)C2)cc1 c1(C(=O)NCC23C(CN(S(CC(=O)OC)(=O)=O)C2)C3)cc(OC)c(O)cc1Br C1(CNC(CN(CCC)C)=O)CC(CNC(C)=O)CN1C(=O)CCNC(=O)OC C(C1CN(C(c2ccc3c(c2)CCO3)=O)Cc2ccccc21)NC(CN(C)C)=O CCC(Cc1cn(CCOC)nn1)C(=O)N1CCOC(c2ncon2)C1 CC(CC(=O)NC1CC(NC(=O)Cn2ccc(O)nc2=O)C1)C(F)(F)C(F)(F)F CN(OCc1ccccc1)C(=O)C1(C)CN(S(=O)(=O)CC#N)C1 N1(C(C(CCOC)NC(c2ccncc2Cl)=O)=O)CCCCCCCC1 N1(C(c2ccncc2F)=O)CCCC(C(N2CCC3(CSC3)C2)=O)CC1 N1(C(c2c(COC)scc2)=O)CC(=O)NC2CN(C(=O)CC3CCCCC3)CCC12 c1(CC)cc(CC)nc(N(CCCNC(C2(n3ccnc3)CCCC2)=O)CC)n1 N1(C(C(C(=O)OC)C)=O)CCC2CN(C(c3cccc(Cl)c3F)=O)CC2C1 c1(C(N2CC(NC(Cc3cn(CC)nc3)=O)C(C)C2)=O)cc2cc(F)ccc2o1 CC1CCC(=CC(=O)N(C2CN(C(c3csc(-c4ncccn4)n3)=O)C2)C)CC1 Cc1ccc2c(C(=O)NC3(C)CCCN(C(c4snnc4C)=O)C3)ccnc2c1 C(C(CN=c1[nH]nc(O)s1)C(F)(F)F)NC(c1c(CC)cccn1)=O CS(=O)(=O)C1CN(C(=O)CC(N)C2CC(F)(F)C2)C2(CCC2)C1 c1(C(N2CCCC(O)(CNC(C=CC(C)C)=O)C2)=O)cc(S(N)(=O)=O)ccc1N C1(N(C(C(C)SCCCC)=O)C)CCCCN(C(=O)C(C)(C)c2cnn(C)c2)C1 C1(C(=O)NCCCC(CO)NC(Cc2c(C)scc2)=O)Cc2ccccc2O1 N1(C(C2C3(CC(NC(CN(C)C(=O)C4CC4)=O)C3)C2)=O)CC(O)(C2CCC2)C1 N1(C(C2(C(=O)OC)CC2)=O)C2CCC1CC(CNC(=O)CSc1nccn1C)C2 N1(C(C2CCC(C)O2)=O)CCC(NC(c2occc2Br)=O)C(F)C1 C12(C(=O)NCC(CNC(c3c(Cl)ccc(OC)n3)=O)O)CC3CC(C(=O)N1)C2C3 c1(CCCC)cc(C(=O)NC(C)CCNC(C2(CO)CC2)=O)c(C)o1 Cc1c(CC(=O)NC2CCC2CNC(=O)C(C)OC2CCOC2)cnn1C C12(NC(c3cccc(C)n3)=O)CCCCC1CN(C(C1(N(C)C)CCC1)=O)C2 c1(C(=O)NCC2CC(NC(c3nc(C(C)(C)C)sc3)=O)C2)ncc(F)cn1 C(=O)(CCN=c1ccc(C)c[nH]1)N1CC(CC=C)(NC(=O)C2=C(Cl)CC2)C1 c1(CC(=O)NC(CNC(c2n[nH]c(C)c2F)=O)C2CC2)ccc(O)c(Cl)c1 C1(CNC(CCCOC(C)=O)=O)CC(C)(C)CCC1NC(=O)CCC=CBr c1(C(=O)NCC(N(C(c2scc(OC)c2)=O)C)C2CC2)cc(C)n(C(C)C)c1C c1(CC)ncc2c(n1)CN(C(c1ncnn1C)C(=O)NC(C)(C)CC)CC2 C1(NC(COC)=O)CN(C(=O)Cc2cnco2)CC2(CC2)C1 C(CCC(C)(C)NC(c1cn(CC(F)(F)F)nc1C)=O)NC(c1c(C)cc[nH]1)=O C1(C(N2C(COC)C(C)(C)C2)=O)CN(C(=O)CCOCC(C)(C)C)CC12CCC2 N1(C(CCn2ccc(C)n2)=O)CC(CNC(c2ccc(Cl)o2)=O)C(O)C1 C12(NC(c3nc[nH]c4nccc3-4)=O)CC3CCC(C1C2)N3C(=O)COCCF N1(C(CCNC(C)=O)=O)CC2CC2(NC(=O)CN2CCOC2=O)C1 c1(C(=O)NC(CC)CN(C)C(C2CCCC2C(F)F)=O)nn(CC)nc1C C(C)(CO)(C(F)(F)F)NC(C1N(C(C(C)CO)=O)CC1)=O CC1CN(C(c2coc(Cl)n2)=O)CC(C)C1N=c1ccnc(C2CC2)[nH]1 C1(NC(c2cnn(C)c2Cl)=O)CCN(C(c2cnc3[nH]ccc3n2)=O)C12CCC2 c1(OC)ccc(F)cc1CN1CCCC(C(c2ccccc2)=O)C1 N1(C(c2ccnc(OC)n2)=O)CCCC(F)(C(N2CCCC(F)(CO)C2)=O)C1 CC1(C)C(CNC(C2CCCN2C(C2(C#N)CC(=O)C2)=O)=O)C1(F)F C1(CCNC(C2(C)CC(C(F)(F)F)C2)=O)CCCCN1C(=O)C(Cl)=CCl C1(CCC(=O)NC(CC=C)CO)CCCCN(C(C2CC(C)(C)CO2)=O)C1 N1(C(c2cnc(C(C)C)[nH]2)=O)CC(CNC(C2(F)CCCC2)=O)C(C)(C)C1 c1(C(=O)NC2CN(C(c3ncc(F)cn3)=O)CC2CO)cccc2ccncc12 c1(C2(CC(C)C)CC2(C)C)nc(C2CCOC2)nn1-c1ccc(Cl)nc1 c1(N(C2CCNC2)C(C2CNC2)=O)ccc(CC2CCNC2)cc1 CCCCC(F)(F)C(=O)N1CC(OC)C(C(=O)NCCc2ccns2)C1 C1(CNC(C2(N(C)C)CC2)=O)(CO)CCN(C(=O)C(C2CCCCC2)O)CC1 C1(C2(NC(CN(CCC#C)C)=O)CC2)CCCN1C(c1sccc1OC)=O N1(CC=CC(=O)NCCCCNC(C2CC(n3cccn3)C2)=O)CCCCC1 c1(OC)cc2c(cc1C(N1CCC(NC(c3cccc(O)c3)=O)C1)=O)CCC2 N1(C(Cc2c(C)occ2)=O)CCC2(NC(=O)CCn3cccn3)CCCC12 c1(C(C(=O)NCC2(F)CCN(C(C(C)CF)=O)C2)(C)C)cccc(Cl)c1F c1(C(N2CCN(CCCNC(C3C(C)C3)=O)CC2)=O)cccc2nccnc12 Cc1c(C(=O)NC(C)(C)CC(=O)N2CCC(N3CCC3)CC2)cccc1O c1(OC)ccc(C)cc1CC(N1CCC(N(C(=O)C(C)CC2CC2)C)C1)=O C1(NC(CNC(CCC)=O)=O)CCC12CN(C(c1ccnc(C)c1)=O)C2 c1(C(C(=O)N(CCN(C(C)C)C(C2CCN(C)C2)=O)C)(C)C)c(F)cccc1F C(=O)(C(O)CC(N)=O)NC(C(=O)NCC(C(C)C)CO)(C)C C(C)(C)(CCC(=O)NC(CN=[N+]=[N-])C(=O)N1CCC(F)(C#N)C1)N(C)C N1(C(c2cc(C)c(O)cc2)=O)CCC(C)(C)C(C(N2CCCC2CC(C)C)=O)C1 c1(C(N2CCC(NC(C3CC(C)C3)=O)C2)=O)cc(C)n(-c2ccc(F)cc2)n1 N1(C(C(C)(CO)NC(C)=O)=O)CCCC(N(C)C(c2ncnc(C)c2C)=O)CC1 c1(C(N2CCC3CCC(C2)N3)C(=O)NC(CC)(C)C)cc2cccnc2o1 C1(OC)CCC(N=c2[nH]c3c(c(=NCC(C)c4ccc(Cl)cc4)[nH]2)COC3)CC1 c1(OC)ccc2c(c1)CC(C(=O)NC1(CO)CN(C(=O)Cc3cscn3)C1)CO2 N1(C(CC2(C#C)COC2)=O)CCN(C(c2ccc(CSC)o2)=O)CC1C C#Cc1cc(CNc2csc(C(F)(F)F)n2)c(OC)cc1F N1(C(C2(CC)CC(C)(C)C2)=O)CC2CCC2(CCNC(c2cncc(N)c2)=O)C1 N1(C(CC(=O)NCC)=O)CCC2(CC2C(=O)N(C)CCOCCCO)C1 C1(CC(=O)NCCC(O)CNC(=O)C=CCN2CCCCC2)(CC=C)CCCC1 CCCCCCCCC(=O)NCC(C)C(F)C(=O)N1CCOC(C)(C2CC2)C1 c1(C(=O)NCC(C)(C2CC2)NC(C2CC(C)SCC2)=O)nc2c(s1)CCCC2 N1(C(CCC(C)OC)=O)CC(CNC(=O)CCc2nccn2CC)CC(C)(C)C1 C=C1Cn2c(C(N3CC(CNC(C4C(Cl)(Cl)C45CC5)=O)C4(CC4)C3)=O)nnc2S1 c1(C(N2C(CCC)CN(C(=O)CC(C)O)CC2)=O)ccc(OC)c(F)c1O c1(OC)ccc(C(=O)NCC(C)NC(=O)Cc2cc[nH]n2)cc1S(N)(=O)=O c1(CC(=O)NCCN(CCC)C(c2cccc(=S)n2O)=O)cc(O)nc(O)n1 C=CC1(CNC(C2OCCC2C(C)C)=O)CCN(C(=O)C=CC2CCC2)CC1 C1(NC(C(C)OCCN(C)C)=O)C2CC3C1C3C2C(N1CCC2CC12C)=O N1(C(c2cn(C)nc2-c2ccoc2)=O)CC(NC(=O)CS(C)(=O)=O)CC2(CC2)C1 C=C(C)CC(C(=O)NOCC1(C)CC1)NC(=O)CC1CCCC(=O)C1 CCC(CNC(=O)C(CCSC)NC(c1cn[nH]c1)=O)(CC)CO c1(COC)nc(C(=O)NC(CNC(C2CC2(Cl)Cl)=O)C2CC2)co1 C(CNC(c1coc(C(F)F)n1)=O)(C(C)(C)C)NC(c1c(C(C)C)c[nH]n1)=O N1(CC)C(=O)NC(c2ccc(Br)cc2Br)C(C(=O)N=c2cc(OC)o[nH]2)=C1C CC(CC(=O)N1CCCC(C)(NC(c2ccc3occc3c2)=O)C1)CC(C)(C)C N1(C(Cc2ccc(C)c(Br)c2)=O)CCC2CCC(NC(=O)CC(C)CF)C12 c1(C(C)C)nc(=NC23CCCC2CN(C(C2(C4CCCCO4)CCC2)=O)C3)s[nH]1 C1(C(N2CC(C)N(Cc3ccccc3)C(C)C2)=O)C2Sc3ccccc3C12 N1(C(C(C=C)OC)=O)CCCC12CCC(NC(=O)CC(C)N(C)C)CC2 C1(C(N(C)CCN(C2CSC2)C)=O)CCCNC1=O Cc1c(C(N)=O)cccc1C(=O)NCC1(NC(C2CC2C2CC2C)=O)CCCC1 c1(C(=O)OC)[nH]c(=NC2CC(CCNC(=O)CC(O)c3ccccc3)C2)sc1C C(=O)(CC(C)(C)C1CC1)N(CCC(N1CC(C(C)C)C1)=O)C c1(CC)nc(C(N2CCC(N(C(C3CC(CCO)C3)=O)CC)C2)=O)cs1 O=C(CCC(CF)CF)NCCSCC(N1CC2CCC(C1)N=C2)=O Cc1nnsc1C(C)NC(=O)C(C1CC1)N(C(=O)Cn1cccc1)C N1(C(C(C2CCCOC2)OC)=O)CCN(C(=O)C=C2CCC2)CC12CCC2 CC(C)(CC(F)F)C(=O)NCC1C2CN(C(c3cncc(C4CC4)c3)=O)CC12 c1(CCNC(C(CN(C)C)NC(CCCSC)=O)=O)cnc(C)cn1 Cn1cc(-c2oncc2C(=O)NCCNC(=O)C(C)(C)c2ccno2)cn1 C(C(C)(C)CCCN=c1nc2c(cnn2C)c(NC2CCC(C(N)=O)C2)[nH]1)OC Cc1c(Br)ccc(C(N2CCOC(C(=O)NCCCn3ccnc3)C2)=O)c1F C#CCCCC(C)C(=O)N1CCC(NC(=O)CCc2cccc(Cl)c2Cl)CC1C N1(C(CC(C)F)=O)CC2(NC(=O)COc3ccc(Cl)nc3)CCC1CC2 C(CS(=O)(=O)C1CC1)NC(c1n(CCCOCC)nnn1)c1ccc(SC)o1 C1(CC)CN(C(=O)CCCc2ccncc2)CCC1NC(=O)Cn1cc[n+](C)c1 C(C)(CCCCNC(C1CCC(C(N)=O)CC1)=O)NC(c1n(CCC)ncc1)=O C1(C(N(C(C)CNC(=O)C(C)OC2CCOC2)CC)=O)CCOC1C N1(C(C(COC(C)C)(C)C)=O)CCC2(CCN(C(C3CCC(C)(C)O3)=O)C2)C1 C(=O)(C(C(C)(C)C)C1CCC1)NC1CCCN(C(c2onc(C)c2C)=O)C1 c1(C(N2CC=CC(NC(Cn3nnc(C)n3)=O)C2)=O)ccc(=O)n(C)c1 CCC(C)C(O)C(=O)NC1CCN(C(=O)COCCOCCO)C(C)C1 N1(C(CCC(C)N(C)C)=O)CCN(C)CC1CNC(=O)Cc1ccc(F)cn1 c1(OC)ncnc(C)c1C(=O)NCCCCN(C)C(c1ccc(O)c(CO)c1)=O C1(CC(=O)N(CC(Cc2ccccc2)C(=O)O)C)COCCOC1 c1(C(=O)NCCC2CCCN(C(CC=C=C)=O)C2)ccc(O)cc1C(F)F CC(C)CCCCC(=O)N1CC(OCCC(N2CCC(CO)C2)=O)C1 N#Cc1cccc(NCC(N2CC3CC(NC(c4coc(Cl)n4)=O)C3C2)=O)c1 CC1OC2(CO)CC1(C(N1CC3CC1CN3C(c1ccc(C(N)=O)cn1)=O)=O)C2 C1(CNC(CSCC(C)C)=O)CCCN(C(C2CCC(O)CC2)=O)CC1 c1(C(C(=O)NC(CC)(C)CNC(c2cnc(C(F)F)s2)=O)C)cccc(OC)c1 Cn1cc2c(n1)CCCC2C(=O)N1CCN(C(=O)C=CC(C)(C)C)C(CCO)C1 C1(C(N2CC3C(N(C(COC(C)=O)=O)C)C3C2)=O)CCn2c(cnc2C)C1 CC(C(=O)N1CCC(O)(C(C)NC(=O)C(O)Cc2cnc[nH]2)C1)S(C)(=O)=O C1(CCC=C)(C(=O)NC(C2(CC)CCC2)=O)CN(C(C2CC2CC(C)(C)C)=O)C1 C#CC1(C(N2CCC(C)(NC(=O)CC(C)SC)C2)=O)CC(=O)C1 C1(C(=O)NC2C(F)CCN(C(CCCCOC)=O)C2)CCn2c(C)cnc2C1 c1(C(=O)NCC2(C)CCC(NC(=O)C3=COCCC3)C2)ccc2cnnn2c1 c1(CC(C(=O)NC(C(C)(C)NC(CCC)=O)C)C)c(C)nn(C)c1C C=C(C)CC(C(=O)NC(CC1CC1)CC1CC1)NC(c1cc(C)c(O)nn1)=O C1(CNC(c2n(CC)ccc2)=O)CCC2(CN(C(c3cncc(N)c3C)=O)C2)O1 CC(O)C(F)(F)C(=O)N1CC(CNC(c2ccc(CCCCO)o2)=O)C2(CC2)C1 C(=O)(C#CC1CCOC1)N(C)CC1CN(C(=O)Cc2cnns2)CCO1 CCCC(C)(CCC)C(=O)NCC1(CNC(=O)C2CCc3nccn32)CC1 N1(C(C(n2ncc(C)c2)C)=O)CC2CC(C1)C2NC(=O)CC1CCCCC(=O)N1 CC(C)CC(C(=O)N1CC(CNC(C2(S(C)(=O)=O)CC2)=O)C(F)(F)C1)N(C)C C#Cc1cccc(C(N2CC(CNC(=O)CSC(C)C)CC2(C)C)=O)c1F N1(C(C(C)C)=O)CCC(C(=O)N(CCC(C)NC(C2(C)CC=CCC2)=O)C)CC1 N1(C(C(CCSC)O)=O)CCCC(NC(c2c(N)cccc2Cl)=O)CC1 Cc1ccsc1C(=O)NCC(C(C)C)NC(=O)CC12CC(c3ccccc3)(C1)C2 c1(OC)cccc(C2CC2NC(=O)C(n2cc(C3CCC(=O)CC3)nn2)OC)n1 c1(C(=O)NC2(c3cccc(OC(F)(F)F)c3)CC2)coc(=O)c2ccccc12 Cc1cc2[nH]c(C(=O)NCCC3CCCN(C(C4CC(C)OC4C)=O)C3)cc2s1 C(=O)(C1=C(Cl)CCC1)NC(CCNC(C(F)=CCC)=O)(C)CC c1(N(C)C)nc(Cl)c(C(N2CCOC(CNC(C3CCO3)=O)C2)=O)s1 N1(C(=O)C#CC2CCC2)CC(C2CN(C(c3sccc3F)=O)C2)C1 c1(OC)ccc(NC(=O)CSC(F)F)c(C(=O)O)c1 CN1CCCC2(CCN(C(=O)COC(S(C)(=O)=O)=O)CC2)C1 C1(CNC(c2c(CCC)nco2)=O)CC2(CCC2)CN1C(=O)COCCCOC C1(NC(=O)Cc2coc(CO)n2)CC2CC1N(C(c1nc[nH]c1C(F)(F)F)=O)C2 C(=O)(CCC(C)(C)C#N)NCCN(C(=O)CCc1ccc(C(F)(F)F)cc1)CC C=CCC(CNC(=O)CC(C)C(C)C)C(=O)NCCCn1ccnn1 C1(C(=O)NCC(c2ccccc2)(C)F)C(C2CC2)C1(F)F C1(NC(C2C(CNC(=O)CC3CC3(Cl)Cl)OCC2)=O)(COCCO)CCCCC1 Cc1nc2ncnn2c(NC(CNC(=O)CCC2(C)CC2)C(C)C)c1C c1(C(N2CC(CCNC(COc3cn(C)nc3)=O)OCC2)=O)csc2nccn12 CC(C)CCC(C(=O)NC1C2CCC(C2)C1CO)NC(C1CC(C(C)C)C1)=O C1(CNC(c2ccn(CCF)n2)=O)CN(C(=O)Cc2cscn2)C2CCCC2O1 C1(NC(c2c(CC)cncc2)=O)CN(C(=O)C(CO)C(C)(C)C)CC1C1CC1 N1(C(COC)=O)CCC2CCN(C(=O)C(c3ccccc3Cl)C)CC2C1 N1(CCC(=O)N(C2CCC(CNC(=O)OC(C)(C)C)C2)C)CCCCC1 CC(C)(C)C(=O)CC(C(C)(C)O)Nc1ccc(OCC(=O)NC(=O)NCC)cc1 N1(CC(=O)N(CCCCC)Cc2ncc(C)s2)CCN(Cc2nnn(C)n2)CC1 CC1CCCC(C)C1NC(C1(NC(C2CCC2)=O)CC(O)C1)=O CCCCCCCC(C)CNCc1cn(-c2c(F)cc(Cl)cc2Cl)nn1 c1(COC(C)=O)nc2ccccn2c1Br.C12CCOC(C1)C(=O)N2C1CC1 C(C(F)(C(=O)NCC1(C)CCCCCC1)C(C)C)NC(C=C(C)C)=O c1(C(N2C3CN(c4nc(COC)nc(C)c4)CC2C3)=O)ccc2c(c1)C(=O)C(=O)N2 c1(NCCCN(C(C2(F)CC2)=O)CC)nnc(Cc2ccccc2)o1 c1(C(N2CCC(C(CNC(CNC(CC)=O)=O)C)CC2)=O)c(N)cc(F)cc1F C1(CC(=O)NCC(CC(C)C)(C)O)CN(C(=O)CC2CCOC2)C2(CCC2)C1 c1(C(=O)NCC(CC=C)NC(=O)C=CC(C)C)ccc(S(=O)(=O)N(C)OC)cc1 C1(CNC(C(C)CC2CCCC2)=O)CC2(CC2)CN1C(=O)C1=NOC(C)C1 C(CC(C)C)(C(=O)N1CCN(C(C2CCSCC2)=O)C(CF)C1)NC(C)=O N1(CC(=O)NCc2ccc(Br)cc2)CC(F)(F)C(F)(F)C1 C=C=CCCCN=c1cc(C)[nH]c(=NCCCCc2ccccc2)[nH]1 c1(C(=O)NCC(CNC(C(CC=C)NC(C)=O)=O)C)ccccc1N=NN(C)C c1(OC(C)C)ccc(N2CC(C(=O)NC(C)Cc3cccc(Br)c3)CC2=O)cc1 C12(C(N(CCNC(CC(CC)CC)=O)CC)=O)CCCCC1CS(=O)(=O)C2 C1(NC(=O)CCc2cnn[nH]2)CC(O)(Cn2cc(CCOCCN(C)C)nn2)C1 C(CC(C)C)(C(=O)NOCCC(F)(F)F)NC(C1CC(C)(CC)C1)=O CC1(C)CC(C(N2CCN(C3CC3)CC2)=O)CN(C(=O)C=Cc2ccncn2)C1 c1(C(=O)NCCC2CN(C(C(C)(C)C3CCOC3)=O)C2)scc2c1OCCO2 n1(CC(=O)NCCCCNC(C2CCOC2)=O)cccnc1=O Cc1ccc2[nH]c(C(=O)NCC3CC3NC(=O)CNC(=O)OC(C)(C)C)cc2c1 Cc1ccc(C(=O)NC23CCN(C(=O)Cc4ccn(C)n4)CCC2C3)c(=O)n1C N1(C(CC(CNC(c2cc(Cl)c[nH]2)=O)OC)=O)CC23CCC2(COC3)C1 C12(C(=O)NCC(COCC)C)C(NC(c3ccsc3C#N)=O)C3CC1C2C3 c1(-c2c(OC)nsc2)ccc(S(=O)(=O)NCc2nccc3ccccc23)c(Cl)c1 Cc1ccc(O)c(NC(C2(CCNC(=O)C(F)C(C)(C)O)CCCC2)=O)c1 c1(C(N2CCC3(C(=O)NC4CC(C)C4)C(C2)C3)=O)cccc2nc[nH]c12 CC(C)CN=C(NCc1ccc(F)c(N(C)C)c1)NC1CCCC(OC(F)F)C1 Cc1oc2cc(C(=O)NC3(C)CN(C(=O)CC4CCC(C)(C)CO4)C3)[nH]c2c1C c1(OC)ccc(OC)c(CC(N2CCN(C(C3CC4CC4C3)=O)C(CO)C2)=O)c1 C(C1c2ccccc2CN1C(C1CC2CC1CC2O)=O)NC(C(CC)C(C)C)=O c1(C(=O)NC2CC(C)(C)N(C(C3CCCCC3O)=O)C2)cc(N)c(F)c(F)c1F CC(C#N)CN=c1[nH]c2c(c(=NCC3(C)CCCC(=O)N3)[nH]1)CCC2 n1(CCCOC)nnnc1C(C1(C)COC1)NC(C)Cc1ccnn1C N1(C(c2c(C)ccnc2)=O)CCC2CCC(C1)N2C(=O)Cn1cnnc1 Cc1oc(CNC(=O)CCn2cccc2)nc1C(=O)NC(C1CCOC1)(C)C CC(C)(C)CCC(=O)N(CCCNC(=O)CNC(N)=O)C1CC1 S(=O)(=O)(c1cccs1)NCC(=O)NC1(CN(C(CC=C)=O)C)CC1 C1(C(=O)NC(C2CCCN(C(c3nccn3C3CC3)=O)C2)C)CSCC(=O)N1 c1(CNC(NOC(C)C)=O)cc(F)cc([N+](=O)[O-])c1 S(=O)(=O)(c1csc(C(N2CCN(C(C3C4COCC34)=O)CCC2C)=O)c1)NC Cc1n[nH]c(C)c1CCC(=O)NC1CC(NC(c2csc(CC(F)(F)F)n2)=O)C1 CC1OC2(CNC(=O)C3CC3)CC1(NC(=O)CCc1cc(F)ccc1Br)C2 C(=O)(C1=NOC(C)(C)C1)N1CC(O)(C(C)NC(c2ncncc2F)=O)C1 c1(C(N2CC3C(CNC(c4scc(C)c4)=O)C3C2)=O)cc(C(C)C)ccc1N C1(OC)(CNC(C2CCCO2)=O)CCN(C(=O)C(=CC2CCCC2)C)C1 N1(C(c2ccc(F)c(Cl)c2)=O)CCC2OCCN(C(=O)C(O)C(F)(F)F)C2C1 N1(C(C2(COCC)CC2)=O)CCC2CCN(C(c3cc(C#N)[nH]c3C)=O)CC2C1 n1(CC)cnc2nc(=NCCC3CC3)[nH]c(NCC3(C(F)(F)F)CCC3)c12 CCCC(C(=O)NC(CN(C(=O)Cc1ccccc1C)C)CC)C(C)C C#CCC(C)C(=O)NC1CCC(CN(C(=O)COc2cnn(C)c2)C)CC1 N1(C(C=CSC)=O)CCN(C(c2ncncc2C)=O)CC(O)C1 C1(NC(C(C)NC(CC)=O)=O)CCCC1Cn1cc(CCC(C)(C)O)nn1 Cc1ccc(C(=O)NC2COCCC2NC(C23CC(C)(CO2)C3)=O)n1C C1(CCCNC(CCOCC(C)(C)C)=O)(CNC(=O)CN2CCCC2)CCCC1 c1(OC)cncc(C(=O)N(CCN(C)Cc2nc(O)n[nH]2)C(C)C)n1 C(=O)(C(C)(C)CS(N)(=O)=O)N(C)CC1COCCN1c1ncc(O)cn1 C(=O)(CCCCC(=O)N1CC2CCC1C(CNC(C13CC(CO)(C1)C3)=O)C2)OC C1(C(N2CC(c3ccncc3)C2)=O)(SC)CN(C(=O)CC2CCCO2)C1 C(c1cccc([N+](=O)[O-])c1)=CC(=O)NC1CCCC(NC(C2(C#N)CC2)=O)C1 CC1CC(NC(=O)CCCCN2C(=O)CCC2=O)CN(C(C2CC=CCO2)=O)C1 C1(CNC(CN(C2CCSC2)C)=O)CCCC(CNC(C2CC(=C(F)F)C2)=O)C1 c1(C(=O)NC(CN(C(c2cc(C)nn2C2CCC2)=O)C)C)c(C)ccnc1O CC1CCN(C(=O)COc2ccccc2)CCN1C(=O)C=CC=C(Cl)Cl CC1OC(=O)NC1C(=O)NCCC1CN(C(c2cc(O)ncn2)=O)C1 C(=O)(C(C)(C)CS(C)(=O)=O)NCC1COCCN(C(CCSCCC)=O)C1 C1(C(=O)NCCN(C)C(C)C)(CC)CCCN1C(C1CN2CCC1C2)=O Cc1ccncc1CC(N1CCCC1C(C)(C)NC(c1nsnc1O)=O)=O C(=O)(C(CCOC)NC(=O)CC(O)C1CCCC1)NCC(=C)C c1(C(=O)NCCNC(Cc2ccc(OC)cc2)=O)ncnc2c1CCC2 N1(C(C2CC2C(F)F)=O)CCN(C(c2cn(C3CCC3)nn2)=O)C(CO)C1 CC1COCCN1CC(C)NC(c1cc(-c2cccc(F)c2)no1)=O c1(C(N2C(CNC(c3cncc(CC)c3)=O)COCC2)=O)cnc2c(c1)COC2 N1(C(C=Cc2ccc(OC)cn2)=O)CC2CCC1CN2C(=O)C=Cc1cnc[nH]1 C1(NC(c2n(C)cnc2)=O)CCCCCC1C(N1CC(S(C)=O)C1)=O Cc1ccc(C(C)C)cc1C(=O)NC1CC(C)N(C(=O)Cc2ccsn2)C1 CC(C)(C)C(C(=O)NCC1CN(Cc2cscn2)CCO1)N1CCCC1=O C1(C(N(C2CCCN(C(c3c(C)cnn3C)=O)C2)C)=O)CCCN(S(N)(=O)=O)C1 C1(CC(=O)NC2CCCC2CNC(c2c(F)ccnc2F)=O)CCC2(CCC2)O1 N1(C(CSCC=C)=O)CCCC(Cn2cc(COC3CCC3)nn2)C1 C=CC1(CO)CCN(C(=O)C2=CCCN(C(=O)CCC(C)SC)C2)CC1 C1(CCNC(CSCCC)=O)CC2CCC(C1)N2C(c1cnc(C(C)C)[nH]1)=O CCC(C(=O)N1CC(F)(F)CC1CCNC(=O)Cc1ccnn1C)C(C)(C)CC C(=O)(C1=CCc2ccccc21)NC1C(CNC(=O)CS(=O)(=O)Cc2cccs2)C1 c1(C(N2CC(O)(CNC(C(C(C)O)NC(C)=O)=O)C2)=O)c(C)nn(C(C)C)c1Cl c1(OC)noc(C)c1C(=O)NCC(CO)NC(C1(Oc2ccccc2)CC1)=O C(=O)(CC(C)CC(=O)N1CCC(NC(C2CC2F)=O)CC1C)OC CC1(C)CCCC(C)(NC(=O)C2=CCN(C(C3(F)CCOC3)=O)C2)C1 c1(OCC=C)ccc(CNC(N2CCC(C(=O)NC)CC2)=O)cc1 Cc1nc(N(c2ncnc3[nH]cc(C#N)c23)C2CNCCOC2)c2sccc2n1 CC1(C)CCC(F)(F)CC1C(=O)NC1CCC1NC(=O)CN=S(C)(C)=O C1(C(=O)OC(C)(C)C)CCC2(CC1)CC(NC(c1ccc(NC(C)=O)cc1)C)C2 c1(C(=O)NCC(C)(CNC(c2n[nH]cc2C)=O)OC)n[nH]cc1[N+](=O)[O-] c1(C(=O)NC(C(=O)NC(c2nnnn2C)C)(C)C)cc(C#N)n(C)n1 C1(NC(=O)Cc2cccnc2)CCN(C(C23CCC(CC2)OC3)=O)CC1O O=CN1CCCC1C(=O)NCCC1CCN(C(C2(c3ccno3)CCC2)=O)CC1 c1(OC)ccc(C(N2CCN(C(=O)CCC3CC(OC)C3)CC2C)=O)c(Cl)n1 C=CCC(C(=O)NC(c1nc(C)oc1C)C)NC(C1CCCC1O)=O C(=O)(C1CCC(=O)c2cccn21)NC1CC(NC(c2nc(C)c(C)s2)=O)C1 C1(C(=O)OCC)(NC(C2CC(NC(=O)C(=CC3CCCC3)C)C2)=O)CCCCC1 N1(C(=O)OCc2cccnc2Br)CC2CCC1C(CN1CCCC1)C2 Cc1c(C(=O)NCC(C)(C)NC(C2CC3CCC2O3)=O)oc(=O)c2ccccc12 c1(C(=O)NCC2(OC)CN(C(=O)C=CCO)C2)c(Br)ccc2n[nH]cc12 CCC(C)CCCC(=O)NCC(COC)NC(c1ccnc2c1CCC2)=O C(C(C)C(=O)NC1CCCC1O)N(C(C=CCC)=O)C c1(NC(C)=O)cccc(CNCCCCCCN2CCCCC2)c1 c1(CC)noc(C(N2CCCC2CNC(C2CCC(=O)N2)=O)C)n1 C(=O)(C(C)(C)C(F)(F)CC)NCCC(=C)CNC(c1cn2ccc(C)cc2n1)=O N1(C(c2c(CCC)occ2)=O)CCN(C(c2cc(C)c[nH]2)=O)C(COC)C1 CC(C)(C#N)CCCC(=O)NC1(C2CN(C(C3CC4CC4CC3C)=O)C2)CC1 C12(NC(CC3CC(OC)C3(C)C)=O)CCC(CC1)N(C(=O)CCCC(C)C)C2 c1(C(N(CCCNC(c2ccc(Cl)c(F)c2O)=O)C)=O)cc2ncn(C)c2cn1 C1(CN(C(=O)C(c2ccc(Cl)cc2)O)C)CCCN(C(c2cnn[nH]2)=O)C1 C1(CNC(c2ccc(C)cn2)=O)CC2(CC2)CN1C(c1cc(N)ccn1)=O C1(C(=O)NCC2(F)CN(C(c3c(CC)[nH]c(=N)s3)=O)C2)CNC(=O)CC1(C)C C(=O)(C(F)C(C)CNCc1nc(C(C)C)cc(C)n1)OCC N1(C(C2CCC(CC)O2)=O)CCCC(C)(CNC(=O)CC2(OC)CCOCC2)C1 C1(NC(c2cc(C)on2)=O)CC2CC1CN2C(=O)Cc1cccc(Br)c1F C1(C(N(CCCC(F)(F)F)C)=O)CC2(CCN1C(=O)CC1NC(=O)NC1=O)CC2 O=C1CN(C(c2noc(C3CCC3)n2)C2CCOC2)CCN1.C1(=O)C(=O)NCCN1 CCCC(C(O)C(=O)NC1(C)CC2(CCC2)C1)NC(C1(C#N)CCCCC1)=O CC(O)C(F)(F)C(=O)N1CC(NC(c2csc(-c3ccoc3)n2)=O)CC(F)C1 C1(C(=O)NCCC2CCN(C(Cc3[nH]c(=N)sc3)=O)CC2)CCOCC12CCC2 c1(-n2c(C(CCCCCC#C)NC3(C)CCC3)nnn2)ccc2c(c1)OCCO2 Cc1cc(OCC(=O)NCC2C(C)CCCN2C(c2cscc2Cl)=O)cc(C)c1 c1(OC)cccc(O)c1C(=O)NCC1CCN(C(=O)C(C)S(C)(=O)=O)C1(C)C C(N=c1[nH]c(=NCC2CCOC2)[nH]c2cc[nH]c12)c1ccc(CC)o1 C1(C(=O)NC2CCN(C(C(C)O)=O)C23CCC3)CCC(C2CCC2)CC1 c1(OC)c(C(=O)NCC2(O)CCN(C(c3cnc(C)cn3)=O)CC2)c(C)nn1C CCCCCCCCC(=O)Nc1cncc(-c2cccc3c[nH]nc23)c1 c1(OC)ncc(C(=O)NCCC(O)CNC(C2(C)CCCS2)=O)cc1C N1(C(C=CCN(CC)CC)=O)CC2CCC1(CNC(=O)C=Cc1cccs1)CC2 Cn1nnc2c(N3CCC(NC(=O)C=Cc4cn[nH]c4)C(F)C3)ncnc12 C1(OC)C(NC(=O)C(C)(C)NC(=O)CC2CC2C2CC2)CC1O C1(CNC(COCC=C)=O)C2CC1N(C(c1ccncn1)=O)C2 Cc1cc([N+](=O)[O-])nn1C(C)C(=O)NC(C)(CNC(C12CC(C)(CO1)C2)=O)C1CC1 C1(C(C2CC3CCC2C3)N(C(CC2C(C)(C)CCO2)=O)C)CCCC2CCCN12 N1(C(c2cn(CCCC)nc2C)=O)CCC(C)N(c2nc3ccccc3s2)CC1 c1(OC)cc(OC)c(C(N2CCC(O)(CCNC(c3ccns3)=O)C2)=O)c(N)c1 c1(NC(C(CC2CCC2)NC(C2C=CCS2)=O)=O)ccc(F)c(O)c1 C1(C(N2CCN(C(C(F)=CC)=O)C(c3ccncc3)C2)=O)CC(C)CC(C)(C)C1 CC(C)C(C(=O)N1CCCCC1CC(N)=O)NC(=O)CSC1CC1 c1(C(=O)NC23CN(C(C(C(=C)C)(C)C)=O)C(C2)C3)cccn2nncc12 Cc1c(C(=O)NCC(C)NC(=O)CC2CCC(O)C2)cccc1C#N N1(C(c2c(C)cccc2)=O)CCCC(NC(=O)COc2cccc(F)c2)C1C CC(C)(CC#N)C(=O)NCCCOCCC(=O)NC1CCCCCC1O C(=O)(C1COc2ccc(Br)cc21)NC1CCN(C(C2(C=C)CC2)=O)CC1F C(=O)(C1=CCC(C)(C)CC1)NC12C(NC(c3ccn(C)n3)=O)CC(CC1)C2 C(=O)(C(C#N)C(C)(C)C)N(C1(C(=O)N(C)CC2CC2)CC1)C.C12(CCCO1)C(=O)N2 N1(C(C2C=CC(NC(C3C(CCOC)C3)=O)C2)=O)CC(N=[N+]=[N-])C1 N1(C(C(CSC)O)=O)CC(C)OC2(CCN(C(c3cccc(C)c3Cl)=O)CC2)C1 N1(C(CC(C)=C(C)C)=O)CCC(C(=O)NOCC2(C)CC2)C1(C)C c1(C(N(c2nc(C)c(Br)cn2)C2CC(N)C2)=O)cc2ccccn2n1 C1(CN(C(=O)C(C2CCCCC2)NC(C2(O)CCSC2)=O)C)CC2(CC2)C1 O=C(C1Cc2ccc(Cl)cc21)NCC1CCN(C(C2CC23CC3)=O)C1 Cc1cc(S(N)(=O)=O)oc1C(N1CCCC(N(C(=O)COC(C)C)C)CC1)=O N1(c2ccnc(SC)n2)CC2CCCN2CC1C c1(CC(N2CCCC(N(C(=O)CCc3ccc[nH]3)C)C2)=O)cc(O)nc(O)n1 C(=O)(CCS(=O)(=O)C(F)(F)F)NCC(CCNC(C=CC(=O)OCC(C)C)=O)O C(C(F)(C(=O)NCC1(CO)CCN(C)C1)C(C)C)NC(C(CC)C)=O c1(CNC(=O)NCCNC(CCC)=O)cn(C2COC2)nn1 C1(C(=O)NCC2CCCN(c3nnc(CCC)s3)C2)CC2(CCC2)CO1 N1(C(c2ccc(F)c(C)c2C)=O)CCC2CCN(C(=O)CC3CCSC3)CC12 CCCC(C)(C)CC(=O)N1CCC(NC(c2cn(C)nc2C(F)(F)F)=O)CC1C c1(CCC(=O)NCC(C)NC(=O)C=Cc2ccc(Cl)s2)cc(F)cc(F)c1 C1(CC(N2C(CNC(c3cc(N)c(Cl)cn3)=O)CC2)=O)COc2ccccc2O1 C1(C(=O)NC2(CNC(c3cccc(CC)c3)=O)CC2)COCC2(CCC2)O1 Cn1cc2c(C(N3CCCC4CN(C(=O)C5=CCCSC5)CC34)=O)cccc2n1 N1(C(c2nc(OC)oc2)=O)CC2CC1(C(=O)N(C1CC1)CC1(O)CCC1)C2 N1(C(C(C=C=C)C)=O)CCC(CNC(c2ccnc(CCC)c2)=O)(OC)CC1 c1(NC(CCCN(C(C)C)C)C)cc(NCC2CCCSC2)nc(C(F)(F)F)n1 C(C(=O)NC(CNC(=O)CCOCC1COC1)C(C)C)(C(C)C)OC(C)C C(=O)(C(O)CCC(C)C)NCC1C(CNC(CCCC(=C)C)=O)C1 N1(C(CCC(C)OCC)=O)CCC2(CC2C(=O)NCC2OC(=O)NC2(C)C)C1 C1(NC(c2nccc(C(N)=O)c2)=O)CCN(C(=O)CC2=CCCC2)CCC1CO CC1CC(NC(c2cnco2)=O)CCN1C(=O)C(F)C(C)(C)O C(CN=c1ccc(C#N)c[nH]1)C1(OC)CN(C(C2CC3(CCOC3)C2)=O)C1 c1(C(CC)(C)C)ccc(CSCCF)cc1.c1(C2(C)CN2)nnnn1C(C)CC C1(NC(CC(C(=C)C)OCC)=O)CC2CC1CN(C(c1ccc(C)c(C)c1)=O)C2 N1(C(CC)=O)CCC(C)N(C(c2cnc(C(=O)OC)s2)=O)CC1 C1(N(C(CCCC)=O)C)CCCC2CN(C(c3cc(C(C)C)n(C)n3)=O)CC12 c1(SC)cc(C(=O)NC(C2(O)CN(C(=O)C(C)(C)c3ccccn3)C2)C)co1 c1(C(=O)NC(c2ccc(CNC(C(C=CC)O)=O)cc2)C)cc(=N)[nH]c(Cl)n1 C1(CNC(=O)Cn2cnnc2O)CC2CCC1N(C(C1C3CCC(=O)C13)=O)C2 Cc1ccc2cc(C(N3CC=CC(O)C3)C(=O)NC(C)(C)C)ccc2n1 CCCC(C)CC(=O)NCC1(CCNC(=O)C(C)CN2CCOCC2)CC1 c1(CCNC(C2N(C(=O)OC)C(C)C2)=O)ccnc2cc(Cl)ccc12 c1(C(N(C2CCN(C(c3c(C#N)ccs3)=O)C2)CCO)=O)c(F)ccc(O)c1F C1(NC(CC(C)F)=O)CC2(CCC(CNC(=O)CCCN(C)C)CC2)C1 N1(C(C2OCCN(C(CCC(C)CN(C)C)=O)CC2)=O)CC2(CCN(C)CC2)C1 n1(C(C(C)C)C)nc(C(c2ccccc2)O)nc1-c1cc(Br)c(Br)s1 Cc1cc(NC(C2COC(CNC(=O)C=CC3CC3)C2)=O)cc(O)c1 C(=O)(CCC(F)(F)F)NC(CC(C)NC(c1coc(-c2ccc(F)cc2)n1)=O)C c1(N(C(C)CCNC(c2ccco2)=O)C)nccc(=NCCC2=CCOCC2)[nH]1 c1(OC)ccccc1C=CC(=O)C(=O)Nc1ncc(C(C)=O)c(C)n1 c1(OCC=C)ccc(Cl)nc1C(=O)NC1COCC1NC(C1(C(C)(C)O)CC1)=O C(CCNC(=O)C(=O)Nc1ccc(Cl)cc1)(C(C)C)NC(C(CC)C)=O c1(C(N2CC(NC(c3ccn(C4CCCCC4)n3)=O)C2)=O)c(F)ccc(Cl)c1F Cc1cc(C(=O)NC(C)(C)CNC(c2c[nH]nc2C(C)(C)C)=O)n2nccc2n1 N1(C(c2cc(CNC(C3C(C)(C)C3)=O)ncc2)=O)CCC2(C1)CC2(F)F c1(C(N2CC3CCN(C(c4c(C)n(C)nc4)=O)C3C2)=O)c(O)nnc2c1CCC2 c1(NC(C)=O)ccc(C(=O)N(C2CCCCC2N(C)C(C23CCC2C3)=O)C)nc1 C1(CC)C(C(=O)NCCn2cc(COC)nn2)CCN1C(c1n[nH]c(O)n1)=O N1(C(c2c(C)cns2)=O)CC2CCN(C(C3C4CCC5C(C4)CC35)=O)C2C1 C1(NC(CCCC)=O)CN(C(c2cn(CCC)nn2)=O)CC1O C(=O)(CCC(=O)N1CCC(NC(C2(C)SCCCS2)=O)C1)N(CC)CC C1(O)(CCNC(COC)=O)CCN(C(C2(C(=O)OC)CCCC2)=O)C1 c1(OC(C)C(=O)NCCNC(C2COC(=O)N2)=O)ccc(Cl)cc1Cl c1(C(=O)NC2CCCCC2C(=O)NCCc2csnn2)c(F)cccc1Cl Nc1c(C(N2CCCC(CCC3CCCNC3)C2)=O)nnc2ccccc12 C1(NC(c2cc(C(F)F)on2)=O)CCOCC1C(=O)NCC1CC2(CCC2)C1 N1(C(C(C)(N(C(=O)CC2CC(C)(C)CO2)C)C2CC2)=O)CCCC2C1CCN2C CC1(C)CCOC1C(N1CC(CNC(=O)CCc2ccc(Cl)nc2)C(O)C1)=O C1(NC(C2C=CCN2C(C2CCC2(F)F)=O)=O)CCC2(CCCC2)C1 c1(OC)ccc(C(=O)CCC(=O)OCC(N2CCC(OCCC3CC3)C2)=O)cc1 N1(C(C(C)=C(CC)C)=O)CCC(C(C)(C)C(=O)NCCC(C)N2CCC2)C1 c1(Cn2cc(C(=O)NC(CCN(C(COCCC)=O)C)C)nn2)ccc(F)cc1 CCCCC(O)C(C)C(=O)NC1CN(C(=O)Cc2cc(F)ccc2F)CC1CC CCCCC(O)CC(=O)N1CC(CCCCNC(c2cnn(C3CC3)c2C)=O)C1 c1(CN2CC(NC(c3c(OC)ncc(F)c3)=O)C(O)C2)c(F)cc(F)cc1F C#CC1(NC(C2CC(NC(=O)CN(C3CCCC3)C)CCO2)=O)CC(F)(F)C1 c1(CCC(=O)NC2CC(NC(C3CC4CC3C4)=O)C2)ccc(C(F)F)cc1 CCC(CC)CC(=O)N1CCC(C(N2CCC(CN=[N+]=[N-])C2)=O)CC1 c1(C(N2CCC(F)(CNC(c3cn(CC)nn3)=O)CC2)=O)cccc2c(C)coc12 C(CNC(C1(CC)CC1(F)F)=O)(CC(F)(F)F)NC(c1ccc(CCC)s1)=O c1(C(N2CCC(CC)C2C(=O)N(C)Cc2cnccn2)=O)cc2n(n1)CCO2 C(c1ccc(OC(C)(C)C)c(OC)c1)=CC(=O)NC(c1cccc(F)c1)CC Cc1cc(C(=O)N(C2CCN(C(=O)CC3(C)CCC3)C2)C)n(C2CC2)n1 N1(C(CCc2ccc(C)nc2)=O)CC(C(N2CCC3(CC2)CC3)=O)CC(F)(F)C1 N1(C(Cc2nc(C)oc2)=O)CCC=C(C(=O)NC2COC3(CCC3)C2)C1 n1(CC)nnnc1C1(NCCS(=O)CC)CC(CCC2CCC2)C1 N(C1CCCn2nccc21)C(C1(CCNC(C(CC)OCC)=O)CCC1)=O N1(C(CN(C2CCC2)C)=O)CCN(C(c2nc(=N)cc[nH]2)=O)CC1CC(F)F N1(C(C(CCOC)OC)=O)CCC2(CC(NC(=O)Cc3c(Cl)cccc3Cl)C2)C1 CC1CC(=O)NCC1C(=O)NCC=C1CCN(C(c2c[nH]c(=N)o2)=O)CC1 N1(C(c2nc(C)cn2C)C(=O)NCCCSC)CC(S(C)(=O)=O)CC1(C)C C(=O)(C(F)C(C)C(F)(F)F)N1C(C)CN(C(=O)C(F)(F)c2cscn2)CC1 C12(C(=O)NCCCC(C)NC(c3c(CC)ncnc3)=O)CC(C)(C1)OC2C N1(C(CSCCNC(=O)NC2C(C)CC2)=O)CCc2ccsc2C1 S(=O)(=O)(c1ccc(N2CCC3(CC2)CC3CO)nc1)NCCCOC C1(CN(C(=O)CC2CCC2)C)CN(C(c2ccnn2CCC#N)=O)CCO1 c1(CN(CC(c2ccsn2)=O)C)ccc(F)c(F)c1F C1(C(=O)NC2(CO)CC3(CCC3)C2)(C(=O)O)CC2(C1)CC(F)(F)C2 c12nc(no1)CC(=O)N2.c1(C)nc(C(C)C)no1.C1(CC=C)(O)CNC1 c1(C(=O)NC(CC)CNC(=O)CC2(C)CCC2)cc(O)nc(O)n1 CC1CCN(C(c2ccc(C#N)[nH]2)=O)CCN1C(=O)Cc1cnc2cccnn12 c1(NC(C2CC(F)CN2C(c2ccc(I)c(F)c2)=O)=O)cc(Br)cnc1F c1(C(=O)OC)cncc(C(=O)NC2CCC(CNC(=O)CSC(F)F)C2)c1C N(C)(S(=O)(=O)N(C)C)CC(N1CC(NC(C=CC)=O)C2C1C2)=O c1(SC)ccc(CCC(=O)NC2(C)CCN(C(=O)C=CC3CCCO3)C2)cc1 N(C(=NCCC(C)C)NCC1(c2ccccc2)CC1(C)C)CCS(=O)(=O)NC C(=O)(C1=C(C#N)CCC1)NC1(COC)CN(C(=O)CCN(c2cnccn2)C)C1 C1(CC(=O)NCCN(C2CCCC2)C(C=CCC)=O)CCOC(C)C1 c1(C(=O)NCC2N(C(C(C(CC)C)(C)C)=O)CCCC2)ccnc(P(C)(C)=O)c1 c1(C(=O)Nc2cccc(CNC(C3(C4CC4)CC3)=O)c2)cn2cccnc2n1 CCCCC(CC)CC(=O)N1CC2(CCN(C(=O)CC3SC(=N)NC3=O)C2)C1 Cc1ncc(NC(C2(C)CCCN2C(c2cc3ccoc3s2)=O)=O)c(Cl)n1 c1(C(N2CC(N(C)C(c3ncoc3C(C)(C)C)=O)C2)=O)cn(C)ccc1=O N1(C(C(CC=C)C)=O)CC(N(C)C(c2cnn(C)c2Br)=O)C2(CC2)C1 C12(CNC(C(CC=C)C)=O)CCC(NC(=O)Cc3cc(F)cc(Cl)c3)(CO1)C2 Cc1nc(C)c(C(N2CC(c3ccccc3)(NC(=O)C(F)C(C)C)C2)=O)s1 Cc1cc[nH]c(=N)c1C(N1CC(O)(C(C)NC(c2cc(Br)cn2C)=O)C1)=O c1(C(CO)N(C)Cc2n(CCC)ccn2)cccc(Br)c1 C(=O)(CC(C)(C)CNC(C1(n2cnnn2)CC1)=O)N1CCC(C)(CC)C1 Cc1ccc(C(=O)NCC23CC(CNC(C4(CC5CC5)CCCO4)=O)(C2)C3)nc1 C(=O)(CCCC(=O)N(C)C)N1CCSCC=C(c2cccs2)C(=O)N1.CC1CCC1 c1(C(=O)NC(C(=O)N2CC(C(CC)CC)C2)CC2CC2)cc(F)cc(F)c1 CC(C)CC(C)C(=O)NC1CCC12CN(C(C13CCC(CC1)CO3)=O)C2 CC(F)(F)C(C)(C)C(=O)N1CCC(CCNC(C2(c3ccsc3)CC2)=O)CC1 Cc1sc(O)nc1C(=O)NC1CN(C(C2CCCN(Cc3cccnc3)C2)=O)C1 N1(C(CSC(C)C)=O)CCC(CNC(=O)Cc2csc(-c3ncccn3)n2)C1 C(C1CCN(C(=O)C(C)N2CCCC2)CC1)=CC(NOCCC(C)O)=O N1(C(c2ccc(CC(N)=O)cc2)=O)CC2(CCCC2NC(c2cnc[nH]2)=O)C1 C1(C(=O)NC2(CNC(C3N(C)CCOC3)=O)CCCC2)CCc2ncsc2C1 c1(OCCNC(=O)Cn2nnc(=O)[nH]2)ccc(F)cc1Cl C(=O)(CCCCCn1cnnn1)NC(C1CN(C(C2CCNC(=O)C2)=O)C1)C C(=O)(CCC(F)F)NCC(COC)NC(CNS(CC)(=O)=O)=O C12(C(N3C(CNC(c4ncc(C)c(C)c4)=O)CCC3)=O)CCCN(CC1)S2(=O)=O C1(NC(c2c(CC)c[nH]c2)=O)CN(C(C2CC3C=CC2C3)=O)CC2(CCC2)C1 N1(C(C2(C#C)CCCCC2)=O)CCN(C(c2nccn3ccnc23)=O)CC(C)C1 c1(OCCC(=O)NCC2CCCC2NC(C2CC3CC3C2)=O)ccccc1Cl c1(C(=O)NC2C(NC(C(C)OCCC#C)=O)CC2)cc(C(C)(C)C)n(C)n1 N1(C(C2(CC)CCOC2)=O)CC2C=CC1C(C(=O)NCCC1CC1)C2 N1(C(C(CC)Nc2nc(C)cs2)=O)CCCc2cc(C(=O)OC)ccc21 CC1CN(C(=O)C(CCOCCO)NC(c2nc(=N)cc[nH]2)=O)C1(C)C c1(C(N(CC(CN(C(C2CN(CC)C(=O)C2)=O)C)O)C)=O)ccc(C)cc1O C1(O)(CCC(=O)NCC2CCCCN2C(=O)C(c2ccncc2)O)CCCCC1 c1(OCC)ccc(S(=O)(=O)NC2=NCCS2)cc1S(=O)(=O)N=c1cc[nH]cc1 CCCC(F)C(=O)NCC#CC(=O)N1CCCC1CO C#CCCC(O)C(=O)N1CCN(C)C(CNC(C2CC(F)(CO)C2)=O)C1 CC(C)C1=NOC(C(N2CCC(C)C(CNC(C3CC=CCC3)=O)C2)=O)C1 c1(C(=O)NC(CCCCNC(CCC(C)OC)=O)C)cnc2c(c1)CCC2 N1(C(C2C(F)(F)C23CC3)=O)CCCC2(CCCN2C(=O)CNC(=O)C(F)(F)F)C1 C1(C(C)O)C(=O)N(c2ccc(N3CCOC(C)C3)cc2)C(=O)N1C C=CCC(C)(CC)C(=O)NCCOCCN(C)C(c1cscc1F)=O CC1=C(C)CC(C)(C(=O)NCC2(C3(O)CN(C(C45CSCC4C5)=O)C3)CC2)CC1 Cc1cc(=O)n(C)nc1C(=O)NCC(C)(CC(C)C)NC(=O)C(C)NS(C)(=O)=O c1(NS(=O)(=O)c2ccc(-c3cncc(O)c3)cc2)ccc(C2=CCNCC2)cc1 Cc1cc(C(N2CC(O)CC2C(N2CC(F)C(F)C2)=O)=O)ncc1N CC(CC(=O)NC(C1(O)CN(C(=O)COC2(C)CCC2)C1)C)P(C)(C)=O N1(C(COc2cccc(C)c2)=O)CC23CCCC2(C1)CN(C(=O)CCC1CC1)C3 c1(C(N(CC(C)N)CC)=O)coc2c(C)cccc12 c1(C(=O)NC(C)(C)CNC(c2ccn(C3CC3)n2)=O)ccc2c(c1)CCCS2 C(=O)(C1CCCc2ncccc21)NC1CCC(CNC(C(C=C)(C)CC)=O)C1 Cc1cnsc1C(=O)NC1(C)CC(C(=O)NCCC2COCCO2)C1 CCCCCC(C)(C)C(=O)NC(CNC(=O)C(O)CC(C)(C)C)C1CCC1 C(=O)(C1CCc2cccc(OC)c21)NC(CC)CNC(CCCC(=O)NCC)=O N1(C(C(C)(C)N2CCC2)=O)CCOCC(NC(=O)C(F)=C2CCC2)C1 c1(C(=O)NC2CN(C(C(c3cncc(F)c3)C)=O)C(C)C2)nccc2[nH]ccc12 C#Cc1cc(C(=O)NCC2(CCNC(c3ccnnc3O)=O)CC2)cc(F)c1 c1(CN(C)C)cc(C(=O)NC(C)(CNC(=O)CC2CC3(CC3)C2)C2CCC2)co1 N1(c2nnc(C(CC)(C)C)o2)CC(NC(c2cnc(C3CC3)o2)=O)CC1C CC1CC(N(C(=O)C(C)(C)CNC(c2ccnnc2)=O)C)CC(C)C1 c1(C(N2CC3C(NC(CCCC)=O)CC(C3)C2)=O)ccnc2[nH]c(O)nc12 c1(NC)nc(C)ccc1C(N1CCC(C)(NC(C2OCCC2C)=O)C1)=O n1(CC(C)NC(=O)C2CC2)cc(CCCC(C)O)nn1 N1(C(c2ccc(CC)o2)=O)CCN(C(C2CN(C)C2)=O)CC2CCCCC12 CCCC(CNC(=O)CCC(C)NC(c1ccncc1O)=O)CCO CCC1=C(C(=O)N2CCC(C(=O)NOCC3CC3)C23CCC3)CCCO1 C(=O)(C1Cc2ccc(F)cc21)O.C=C(C)C(C)(C)C(=O)N1CCC(O)(C)C1(C)C(=O)OC c1(OC)ccc(C(N2CC(CN(C)C(c3cc(Cl)sc3Cl)=O)C2)=O)cn1 Cn1ccc(C(=O)N(CCC(=O)N(CC(C2CCC2)CCO)C)CCCO)c1 C(=O)(C(CCCO)c1ccccc1)NCC1(NC(=O)CN2CCCS2(=O)=O)CC1 Cc1ccc(OC(C)C(=O)NCC(O)CNC(c2cc(CN(C)C)on2)=O)cc1 c1(C(N2CC(N(CC(C)C)C)C2)=O)conc1C(C)NC(c1nnsc1N)=O C1(C(=O)OCC)OCCOC1C(=O)NCCCCn1cc(COC(F)(F)F)nn1 c1(N2CCC(CNC(c3c(C)nc(CO)s3)=O)C23CC3)ncnc2scnc12 C(c1cc(Br)cs1)=CC(=O)OCCOC1(CC(C)=O)CCCC1 c1(OC)cncc(CNC(=O)C(C)C(C)NC(=O)CN2CSCC2=O)n1 C1(NC(c2c(C)con2)=O)CC(NC(c2nc(C(F)(F)F)cn2C)=O)CC1O c1(C(=O)NCCC(CNC(C2CCC2C)=O)OC)ccncc1F c1(C(=O)NC2C(NC(C3CC(OC(C)(C)C)C3)=O)C2)[nH]cc2c1CCS2(=O)=O C(=O)(Nn1ccccc1=O)c1cnc(CNC(C(C)C2CCC2)=O)nc1 C1(CCCCNC(C=CCC)=O)CCN(C(=O)COC(F)F)CC1 c1(C(c2n(CC(=C)C)nnn2)NCc2ccc(Br)cc2Cl)cccc2cncn12 N1(CCNC(CCC)=O)CCCN(C(=O)CCC2(C)CC2(F)F)CC1 N1(C(C(C)C(C)O)=O)CC2CCC(C1)C(NC(c1cc(N3CCCC3)ncn1)=O)C2 N1(C(c2occ(OC)c(=O)c2)=O)C2CCC1CN(C(=O)C1=CC3CCCC13)C2 c1(NC(C(CNC(c2c(CCC)nco2)=O)N(C)C)=O)ccc(OC)c(CC)c1 n1(CCNC(C(c2cccs2)NC(C(CC)NC(N)=O)=O)=O)ncccc1=O c1(CC)cc(C(=O)NC(C)CN(C(=O)CCc2nnc(S)nc2O)C)c(C)nn1 CCC(C)C(=O)N1CCCC1C(=O)NCc1nccs1 c1(-n2c(C(C3(C(C)CO)CC3)NC(C=C)(C)CC)nnn2)ccc2c(c1)CCC2 C(C(=O)N1CCCCC1CN(C)C(c1cnsc1)=O)(C(C)(C)C)NC(C)=O Cc1cc(C)n(C(C)CC(=O)NCC2CCN2Cc2nccs2)n1 c1(CC)ccc(C(N2CCCC2CNS(C)(=O)=O)C(=O)NC2CCOC2)cc1 CC1(C(=O)NCCN(C2CCCCCC2)C(c2n[nH]cc2Cl)=O)CCC(=O)N1 c1(C(N(C2CCN(C(c3c(SC)nn(C)c3)=O)C2)CCO)=O)nccc(C)c1N N1(C(c2scc(OC)c2)=O)CCC2CN(C(=O)Cc3cc[nH]n3)C2C1 N1(C(Cc2n(C(C)C)cnn2)=O)CCCC(N(C)C(c2cc(F)n(C)n2)=O)CC1 c12ccc(Br)cc1NC(=O)NCCCOC2=O.C(=O)(N(C)C(C)C)NC CC(C(=O)NCCCNC(c1[nH]c(=N)ccc1Br)=O)C(C)C(C)(C)C c1(NC(C)=O)ccc(NC(=O)CN2CCC(NC3CCCC(O)C3)CC2)cn1 c1(CCC(=O)NCCCNC(=O)CC23CCC(CC2)C3)nc2ccccc2[nH]1 Cc1ccc(C(=O)NCC(CO)NC(C2CCCN2C)=O)cc1NS(C)(=O)=O N1(C(C(c2scc(C)n2)C)=O)CCCC(NC(c2cc(C(C)C)on2)=O)CCC1 C(=O)(CCC(F)(F)C(F)(F)F)N1C(C)CC(NC(C2(CCO)CC2)=O)C1 Cc1ccc(CCC(=O)NC2CC(NC(c3c(C)ncn3C)=O)C2)cc1Cl C(N=c1[nH]nc(C(F)F)o1)C1CCCN(C(c2cn(CC(C)C)nc2)=O)C1 CN1CCN(C(=O)CCC2CCN(Cc3cccnc3Cl)CC2)CC1C(=O)O Cc1cnc(CN2CCC(O)C2C(=O)NCC(N2CCOCC2)=O)cc1Br CN1CC(NC(c2conc2CNC(C2CC3(CCC3)CO2)=O)=O)C(F)(F)C1 C1(CNC(C(C)C#N)=O)CN(C)CCN1C(c1cc2ccsc2s1)=O CC1C(NC(=O)CC2CCCOC2)CCCN1C(=O)CCS(N)(=O)=O C1(C(N(CCCNC(c2cc[nH]c2)=O)C)=O)CCCC(C(F)F)C1 N1(C(CCOCC)=O)CCCC(C(N2CCCC2c2ccncc2)=O)C1 N=S(=O)(CCNC(c1ccccc1[N+](=O)[O-])=O)c1ccc(Br)cc1 N1(C(C2(OC)CCC2)=O)CCC(C(N2CC3(CCC3O)C2)=O)CC1(C)C C(=O)(CCCS(N)(=O)=O)N1CC2CC(NC(c3ncc(OCC)nc3)=O)C2C1 c1(CN2C(C)(C)CN(C(C3CCCNCC3)=O)CC2)c(Br)cc(F)c(F)c1F C12(C(=O)NCC(C)CN(C)C(C3COCCOC3)=O)CCC(CC1)CC2 CCS(=O)(=O)CCNC(=O)CCC1CCCN(C(=O)CC2CCCN2C)C1 c1(C(=O)NC(CC)CN(C(=O)C(=Cc2cn(C)cn2)F)C)cn(C)c(=O)c(C)n1 CC1(C2CCC2)CCN(CC(O)CC2(O)CCCCC2)C1.C(CC#N)N c1(C(N2C(CCNC(c3n(C)cnc3)=O)CCC2)=O)c(Br)ncn1C C1(C(N2CCC(Br)C2)=O)C2CC1N(C(c1ccccc1-c1cnco1)=O)C2 CC1(C)CC(CN)N(C(C2CS(=O)(=O)CCO2)=O)C1 C12(CNC(c3nc(OCC)sn3)=O)CCC(CC1)N2C(C1CCC(CC)O1)=O C#CCC(C(=O)NCC(C)(C)CN(C(c1ccc(C(=O)OC)cc1)=O)CC)C1CC1 C(CCC(c1nnnn1C1COC1)(C1CC1)NCC1CC12CC2)OC CC1CCN(C(c2ccoc2Cl)=O)C(CNC(c2nccnc2C(N)=O)=O)C1 c1(CSC)ccc(C(N2CC(Cn3cc(CC4(O)CCC4)nn3)C2)=O)o1.S(C)(=O)(=O)N N1(C(c2c(CC(=O)OC)occ2)=O)CC2(CCC2CNC(=O)CNC(C)=O)C1 CCC(C)C(C)CNC(=O)C(c1ccco1)NC(=O)C=Cc1nccs1 C(=O)(C1OCCc2ccc(C)cc21)N(CCN(C(C(CCC=C)(F)F)=O)C)C c1(CC)nnc2cc(N3CC(NC(C45CCCCC4C5(F)F)=O)C(C)C3)ncn12 Cc1cc(NC(c2sc(NC(c3ccc(C(=O)OC)cc3)=O)nc2C)=O)n(C)n1 C1(C(=O)NC(C)COC(F)(F)F)CC(NC(c2ncncc2Cl)=O)C1(C)C c1(C(N2CC(F)(CNC(=O)C(F)=C3CCCC3)C2)=O)nc(O)nc(O)c1F C(CC(C(=O)N(C)Cc1cncn1C)NC(C1CC(OC)(OC)C1)=O)=CC c1(C(=O)NC2CN(C(CCS(N)(=O)=O)=O)CC(O)C2)cc2ccc(Cl)cn2c1 c1(CNC(C(C(C)OC)NC(CCC#CC)=O)=O)c(O)cccc1F CCCC(CC)CC(=O)N1CC(NC(=O)Cc2csc(-c3ccsc3)n2)C1 c1(SC)ccc(CC(C2(CNC(C(Cc3ccoc3)N)=O)CCCC2)=O)cn1.SC C1(N(C)C)(C(N)=O)CCN(C(c2ccnc(Cl)c2F)C(=O)NCCC2CC2)CC1 C(CCCCCCC)NC(C1(CC=C)CCN(C(=O)CCCC(=O)OC)C1)=O C(=O)(C1=C(Cl)CCOC1)NCCCCCN(C(C(CC)SC)=O)C Cc1cc(C(=O)NCC2(O)CC(NC(=O)CCC(C)N(C)C)C2)ccc1Cl C12(C(N(CCn3cncn3)CC)=O)CCC(NC(=O)OC(C)(C)C)(CC1)C2 [N-]=[N+]=NCCCC(=O)NC1CCCCC1CNC(=O)CC(c1cccc(F)c1)O CC1(C(=O)NCCNC(c2ccc(OC(F)(F)F)nc2)=O)CC2C=CC1C2 C1(CNC(C2C(C)C2)=O)CCN(C(c2ccccc2NS(C)(=O)=O)=O)CC1(F)F CCC(C)C(O)CC(=O)N1CCC(F)(C(=O)NC2(c3ncc[nH]3)CC2)C1 C(C(C)(C)CN=c1ccnc(NCc2ccnc(OC(C)(C)C)c2)[nH]1)N(C)C C=C(C)CCC(C(=O)Nc1ccc(Cl)cc1F)N1CCC(Oc2ccccn2)C1 c1(CCC(=O)NCCN(c2ccccc2)C)ccc2cnn(C)c2c1 n1(CC(=C)C)nc(COC)nc1-c1cc(C(F)(F)F)ns1 CC1CN(C(C2SC3C=CC2CC3)=O)CCN1C(c1ccc(CCO)cc1)=O CC(O)C(F)(F)C(=O)NC(C)CC1CN(C(=O)C(c2cccc(F)c2)O)C1 c1(CC)ccc(C(=O)NCC(C)(C2CC2)NC(=O)Cn2cnnc2)cc1Cl c1(OC)ccc(C(=O)NCC2(CO)CCN(C(C3CC(C)(C)CO3)=O)C2)c(C)n1 c1(C(=O)NC(CN(C(c2ccon2)=O)CC)C)cc(F)cc(N)c1F c1(C(C(=O)NCC2CC2)N(CC)Cc2ccoc2)csc(Br)c1 S(=O)(=O)(c1ccc(OC(C)C)c(C)c1)NCc1c(C(=O)OC)c2c([nH]1)cccc2 C(=O)(CC(CC)C(C)C)N1CCC(CC=C)(C(=O)OC)C1.N12CC(C)C(C)(C1)C2 O=C(C(O)C(F)(F)F)NC(C(=O)NCC1CC12CCOCC2)C1CCC1 C12(C(N3CC(NC(=O)NC)C3)=O)CCCC1N(C(=O)Cc1csnn1)CC2 S(=O)(=O)(c1c[nH]ccc1=NCCCC1CCOC1)NCC(CCC)(C)C CC(C(=O)NCC(CC1CC1)C(=O)NC1CCN(CCCO)C1)S(N)(=O)=O Cn1nc(CNC(C2CC(=C3CCC3)C2)=O)cc1C(=O)NCc1ccncc1Cl CC1CCCC=C1C(=O)NCC(C)C(F)C(=O)NCCCc1ccco1 c1(C(=O)NC(CNC(C(CC)COC)=O)(C)CC)cc([N+](=O)[O-])n[nH]1 N1(C(c2c(SC)cccc2)=O)CCC(C)(CNCc2c(Br)ccnc2Cl)CC1 Cn1nc2c(c1NC(c1sccc1NS(=O)(=O)CCBr)=O)CCC2 C1(NC(C(C)(C)C2CCOCC2)=O)COCCN(C(=O)Cc2csnn2)C1 CC1CN(C(=O)C(C)(C)n2cccn2)CCN1C(C1CCN(C)C1)=O N1(C(Cc2c(NC(C(c3ccccc3)OC)=O)cccc2)=O)CC2CCCCC2C1 c1(C(N2C(CNC(c3ccc(C)nc3)=O)C=CC2)=O)ncc(Cl)cc1O N1(C(c2ccn(C3CC3(F)F)n2)C(=O)NC(CC)C)CCN(C)CC1(C)C N1(C(CC2(N(C(C3C(CCOC)C3)=O)C)CC2)=O)CCCC1c1ncc[nH]1 C1(NC(CCc2cc(C)sc2C)=O)CN(C(C2CC2CC(C)C)=O)CC2(CC2)C1 C(=O)(C(CC(C)C)OC)NCCC(=C)CNC(c1ccc(F)cn1)=O C(=O)(C(C)C(C)C(C)(C)C)OC.N12CCN(CC1)C(=O)CCC13CC(C1)(C3)C2=O c1(CNC(C(Cc2ccco2)NC(=O)CCc2cnoc2)=O)ccc(F)c(O)c1 N1(C(C2CC(CC)NC(=O)C2)=O)C2CCC1CC(NC(=O)CN1CCOCC1)C2 CCCCC(C)C(=O)NCCCCC1CN(C(=O)C=NOC)C1 N1(C(C(=O)NCC2CN(C)C(=O)C2)=O)CCCC(C2CCOCC2)C1 c1(C(N2CCC(C)C2CNC(=O)CCC(N)=O)=O)csc2nnsc12 C1(C)(C(N(C)CC2CCCN2C(c2ccc(F)o2)=O)=O)COc2ccccc2O1 C=C(C)C1OCCC1C(=O)N(C(CC(F)F)C(=O)NC(c1ncc[nH]1)C)C c1(OC)ccc(CC(=O)OCC(=O)Nc2cccc(I)c2)cc1[N+](=O)[O-] CC1=NOC2(C1)CC(C(N1CCCC(CO)(CNC(c3ccsc3Cl)=O)C1)=O)C2 c1(CCNC(C(C)OC(c2ccc(C)cc2C#N)=O)=O)ccc(Br)cc1[N+](=O)[O-] c1(CCNC(=O)NCC2CCCC(N(C)C)C2)nc2c(s1)CCCC2 C(=O)(C(C)C(O)CC(C)C)NC(CC(=O)NC(COCC)C)CC(C)C N1(C(COC2CC(NC(C(CC3CC3)OC)=O)C2)=O)CC2(COC(=O)N2C)C1 c1(OC)cc(C(=O)NC2CN(C(c3nn(C)c(C)c3Br)=O)C2)ccc1C#N C(c1ccc(Cl)cc1)=CC(N1CC(NC(C(C)C2CC2)=O)C(C)C1)=O C1(NC(COC2(C#C)COC2)=O)CC12CCOCC2 c1(C(=O)NC2CN(C(COCC)=O)C(C)C2)cc(NS(C)=O)ccc1F c1(SC)cc(C(=O)NC2(CF)CCN(C(C3(C)CC(C#N)C3)=O)C2)oc1C C(CC(C)C)(CC(C)C)NC(C(C)NC(C1C(OC)CCC1)=O)=O C(=O)(C(C(C)C)NC(c1ccnc(C)c1)=O)N1C(CCCC)CCC1 c1(CCC(=O)NC2C(NC(C(C)c3ccsn3)=O)CC2)ccc(Cl)cc1 Cc1nc2c([nH]1)CC(C(=O)NC1CCCC1NC(c1ccc(Cl)c(O)c1)=O)CC2 c1(NC(CC(CNC(=O)Cc2ccc(C)nc2)OC)=O)ccc(F)cc1C S(=O)(=O)(c1cccc(=NCCCF)[nH]1)NC(c1ncccc1C(F)(F)F)C Cc1cc(C(=O)NCC(C2CC2)N(C)C(c2ccsc2)=O)cc(Cl)n1 c1(C(N(C)CC2(CNC(C3(C=C)CC3)=O)CC2)=O)cnc(O)c(OC)c1 c1(CC)ccc(C(=O)NC2(CCNC(=O)C(C)CSC(F)(F)F)CCC2)c(N)c1 c1(C(=O)NCC(C2CC2)NC(CNC(CC)=O)=O)cnn2c1S(=O)(=O)NCC2 N1(C(C(C(C=C)C)C)=O)CCn2ncc(CNC(=O)Cn3nccn3)c2C1 C1(NCc2cnc(=N)[nH]c2)CCOCC12CCC2 c1(NC(=O)CC(O)C2CCCC2)ccc(NC(=O)Cc2ccsc2)cc1 N1(C(C=CCC)=O)CCC(F)(CNC(c2ccc(C3CCC(=O)N3)cc2)=O)CC1 c1(CN2CC(CC(=O)Nc3cccc4c3CCO4)OCC2)cc(F)c(Cl)c(F)c1 CC(C)(C(=O)N1CCCOC(CNC(C2(C)CC=CCC2)=O)C1)C(F)F C(C(CC(C)C)C(=O)NC(C)CC1CCOC1)NC(Cc1c(C)ocn1)=O N1(C(CCC=C)=O)CCC2CC12C(=O)NOCC(C)C c1(OC)ccc(C(=O)NCCCNC(=O)CCCOc2ccccc2)c(F)c1 C1(OC)CN(C(C2CCCCN2C(c2cc(C)ccc2C)=O)=O)C2(CCCC2)C1 C(=O)(C(CSC(C)(C)C)NC(=O)OC)NC(CC)COCC(F)(F)F N1(C(c2c(C)nc(CCCC)s2)=O)CCCC(NC(=O)CCNC(C)=O)C(F)C1 N1(C(CC)=O)CC2CN(Cc3c(C)nn(C)c3C)CC12 C1(CC=C)(NC(c2scnc2C)=O)CCN(C(=O)CC2CCCCC2C)CC1 c1(C(N2CCCC(c3ccc(F)cc3)C2)C(=O)NC)cccnc1O C1(C(=O)NC(C(C)C)CNC(=O)CCN2CCOCC2)CCCOCC1 C(=O)(CC(F)(F)F)N1CCC(n2cc(CCn3ncc(C(N)=O)c3)nn2)C1 c1(-c2nc(-c3scc(C)n3)nn2CC(F)F)cn2cccc(C)c2n1 C#CC1(C(=O)NC23CCCC2C3)CCN(C(C23CC(CO)(C2)C3)=O)CC1 C(=O)(C(F)CCC(C)C)NC(CC)C(=O)NCC=CBr c1(C(=O)NCC(CNC(c2ccn(C(C)(C)COC)n2)=O)OC)ccoc1C C1(C(N(C)CC#N)=O)Cc2c([nH]c3ccccc23)CN1Cc1cc(Br)ccc1Cl c1(OC)cc(C)c(C(=O)N(C2CCN(C(=O)Cc3ccc(C)c(Cl)c3)C2)C)cn1 c1(C(N2C(C)(CC(=O)NC(C#C)CC)CC2)=O)cccc2[nH]ncc12 N1(C(c2cnc(OC)nc2)=O)CCN(C(C2(C)CC2(C)C)=O)CC(C)(F)C1 c1(CC)c(C(=O)NCC(C2CCC2)NC(=O)C=CC2CCCN2C)cnn1C C1(CNC(C(N(C)C)C2CC2)=O)CC2(CO1)CN(C(=O)Cc1sc(O)nc1O)C2 c1(OCC(N2CC(NC(CC(=O)N(C)C)=O)(CO)C2)=O)ccccc1C(C)(C)C C(=O)(CN=c1cc[nH]cc1)NC1C(C=C)CN(C(=O)C(=O)CC(C)CC)C1 C1(C(=O)NC(c2ccccc2F)C)C2CN(C(c3cccc(Cl)c3)=O)CC12 c1(CNC(CC2(CNC(C(N3CC(C)C3)C)=O)CC2)=O)cnc2n1CCC2 CC(CF)C(=O)N1CCCC1C(C)(C)NC(=O)CC1CC1 CCCCCCC(C)C(=O)NCC1CCN(C(=O)C(CC(C)C)N(C)C)CC1 c1(C(=O)NC2CC(n3cc(C(C(C)(C)C)O)nn3)C2)cccc2c1OCCCO2 C(C(O)CN=c1c(C)c[nH]cc1[N+](=O)[O-])NC(CCc1cc(OC)no1)=O Cc1cnnc(NC(CS(C)=O)C(C)(C)C)c1C#N C(C(C)(C)CC(=O)N(CCC(=O)NOCc1cccc(C)n1)C)OC N1(N(C)C(C23CC(C)(C2)C3)=O)CCC2(CC1)CC2c1cn(Cc2cccs2)nn1 C(C)(N=c1[nH]c2c(c(=NC(C)c3nncs3)[nH]1)COC2)c1nc(C(C)C)[nH]n1 C1(C(=O)N(CCN(C)C(c2cnc(C3CC3)s2)=O)C(C)C)(OC)CCCC1 c1(C(N2CCOCC(C(N3CC(SC(F)F)C3)=O)C2)=O)cc(F)cc(F)c1 N1(C(=O)CCCCBr)CCC(C2CN(C(c3ccc(I)cc3[N+](=O)[O-])=O)C2)CC1 CCCC(C(=O)N1CC2CC(CNC(c3cn(C)[nH]c3=N)=O)C2C1)C(C)C N1(S(CC)(=O)=O)CC2CCCCC2(CN=c2cc(C(COC)OC)nc[nH]2)C1 N1(C(C(CCC)OC)=O)CC2(CNC(=O)C(C#N)C(C)(C)C)CCC1CC2 c1(OCC)ccc(-c2ccc(C(=O)Nc3ncc(C)s3)nc2)cc1OC C1(C(=O)NCC2(CO)CCN(C(COCCN(C)C)=O)C2)CC(C)(C)CN1C N1(C(C)=O)CCNC(=O)C1CN(C1CC2(C1)CC(CO)C2)C(=O)CSCC(=O)O C1(C(N2CC(F)(CC)C2)=O)CN(C(c2n[nH]cc2Cl)=O)CC1F CCC(CC)C(C(=O)NCC(CNC(c1cccc(C(F)(F)F)c1)=O)OC)OC CC(C1CCCc2cccnc21)NC1CCS(=O)(=O)C(C)C1 n1(CCC)cc(C(=O)NC(C2CCOC2)CNC(C2(Cl)CC2)=O)nn1 C1(C(=O)NCC(C)CN(C)C)CCCN(C(c2ccnn2C(F)F)=O)C1 C=C=CC(C)C(=O)NC(C)(C)CN(C)C(c1cn(C)cn1)=O Nc1ccc(C(=O)NC(CNC(=O)C=Cc2cccnc2)C2CCC2)c(O)c1 Cc1ccc(C(N2CC(CC(F)C(=O)NC3CCC(F)(F)C3)C2)=O)nn1 C(CC(C(=O)NCC1(C(C)C)CCOCC1)NC(C1C2CCC(F)C12)=O)OC C1(CNC(C=CCN(CC)CC)=O)CCCCN1C(=O)COC1CCCC(C)C1 c1(C(=O)NC2COCCN(C(C3(C)CC(=C)C3)=O)C2)cccc2c1NC(=O)CO2 C#CC1(C)CCCN(C(C23CCCC2CN(C(C2CS(=O)C2)=O)C3)=O)C1 c1(C(=O)NCCCN(C(=O)C#CC2CCOC2)CC)nc[nH]c2ncc(Br)c1-2 c1(N(c2onc(C(=O)OC)c2C)C)ccc(-c2ccccc2)cc1OC CC(C)(C)CC(C)(C)C(=O)NCCC1(O)CCN(C(c2cnncc2O)=O)C1 C(=O)(C(C)(F)C(=O)OC)N1CC(NC(c2cc(CC)n(CCO)n2)=O)C1 N1(c2nc(C(F)(F)F)cc(C)n2)CCC2(CC1)OCCC2NC(C1CC1(C)C)=O O=S(=O)(c1c[nH]ccc1=NCC1CC(O)C1)N1CCC2(CC1)OCC1CC21 N1(C(CCOC)=O)CCC2(CC1)CC(NC(C1CCc3cn(C)nc3C1)=O)C2 Cc1cccc2c(C(=O)N(C)Cc3cnc4ccccn34)n[nH]c12 c1(-c2occ(CN(C)Cc3cnn(C(F)F)c3)n2)c(Cl)cccc1Cl Cc1nc2cc(C(=O)NC3CC(CNC(=O)CCC(F)(F)F)C(O)C3)cnc2s1 C1(CC(=O)NC2COCCC2NC(=O)C2=CSCS2)CN2CCN1CC2 N1(C(CCCOCC)=O)CCC(CNC(=O)CC(C)n2ccnc2)(OC)CC1 C1(OC)CCn2cc(C(=O)OCc3nn(C)cc3Cl)nc2C1 c1(CN2C(=O)CCC(c3n(C)nnn3)(NC3CC3)C2)cc(P(C)(C)=O)ccn1 N=c1[nH]c2ccc(C(=O)NCCN(C(=O)CCc3nncs3)CC3CC3)cc2o1 CC1(C)CCC(N=c2[nH]c(=NCc3ccc(C(F)F)c(F)c3)c3[nH]ccc3[nH]2)C1 c1(CN2CCC(N(C(=O)CCN3CCCCC3=O)C)CC2)c(N)cccc1F C(=O)(CCCCCN=[N+]=[N-])N1CC(C#C)N(C(c2cnccc2Cl)=O)CC1 C1(C(N(C(C#C)C2CCC2)C)=O)CCN(C(c2sccc2CC)=O)C(C)(C)C1 c12cccc(c1F)-c1nc(cs1)NC2=O.c1(SC)c(C)ccnc1C C1(C(=O)NCCN(C(C2(c3cccc(F)c3)CCC2)=O)CC)CCCC(C)C1 CCCC(C)(O)C(=O)NCCCCCCN(C)C(c1c(C)ccnc1O)=O C1(NC(c2cncnc2)=O)CN(C(=O)Cc2cc(Cl)cs2)CC1n1cccn1 C1(NC(c2c(C(C)C)ncs2)=O)CN(C(C2CCC(N=[N+]=[N-])C2)=O)CCC1C n1(-c2cccc(C)n2)ncc(=NC(=O)NCC2CCOCC2O)[nH]1 c1(C(N2CCC(NC(=O)CCC3CC3)CC2C2CC2)=O)cc(F)c(F)c(O)c1F c1(C(N(C2CCCCC2)C)=O)ccc(NC(=O)Cc2sncc2Br)cc1 c1(C(N(CC(=O)OCC)CC=C)=O)csc(CNC(=O)Cn2cccc2)c1 C1(O)(CC#C)CC(C(=O)NC2CC2CNC(c2ncsc2-c2ccccn2)=O)C1 C1(OCCC)CCCCC1C(=O)NCCCC(C)(C)NC(c1nc(=N)cc[nH]1)=O Cc1ccc(CC(=O)NC2(CCCNC(C34CCCN3CCC4)=O)CC2)cc1F Cc1ccc(-n2cc(CN)nn2)c(Br)c1.C1(C(=O)NCCO)CC(=C2CCC2)C1 CCC(CCC(=O)N(C(C)CC(F)(F)F)C)NC(C1C2CN(C)CC12)=O c1(OC)cc(CO)ccc1C(=O)NCC(CC(C)C)NC(c1ccc(F)cc1)=O C1(C(=O)NCc2n(CC)cnc2)CC(NC(C2(C(=O)OC)CC2C)=O)CCO1 CC(C)C(C)C(=O)N(CCCCN(C(=O)CC(C)NC(c1ccccc1)=O)C)C Cc1cc(C)c(C(=O)NC2CN(C(=O)CSc3cccc(Br)c3)C2)c(=O)o1 C1(N2CC3C(CC)(C3)C2)CC2CCC(C1)C2 c1(C(N(CCCCNC(CC(C)OC)=O)C)=O)cc(S(C)(=O)=O)cs1 CN(CCc1cccc(O)c1)N1CCCCC1Cc1cccnc1 S(=O)(=O)(c1ccccc1)N1C(C)(C(=O)NC2C(C(=O)OC)C2)CCC1 N1(C(c2cnn(C(C)(C)C)c2Cl)=O)CC(NC(C2(C)CCNC2=O)=O)CC(F)C1 C1(CC(=O)NCc2cn(CC)nn2)CC2(CC2)CN1C(c1ccc(C#N)cc1)=O c1(NC(C)=O)nc(C(F)(F)F)oc1C.c1(C(N2C(C)C2)=O)n[nH]cc1C(F)(F)F c1(C(=O)NCC(=O)NC2CC(CNC(CC3C(C)(C)C3)=O)C2)ccccn1 C(=O)(CC(C)CC(C)C)NC1C(NC(C(c2ccc(OC)c(F)c2)C)=O)CCC1 c1(NC(C)=O)c(-c2ccccc2)sc2ccccc12.N12CC3C(C3C1)NC2=O Cc1cnc(-c2cn(C(C)C(=O)N(C3CC(OC(C)(C)C)C3)CC)nn2)c(C)c1 c1(CN2CCN(CC(=O)NCCC(C)C)C(=O)C2)cc(F)c(O)cc1F C1(NC(c2c(SC)n(C)nc2)=O)CCN(C(=O)C(C)(C)CF)CC1CO N1(C=O)CC23CCCCC2(COC3)C1.C1CC2CCCC(C1)C2 N1(NC(C(C(C)CC2CCOCC2)N(CCCF)C)=O)Cc2cccc(Cl)c2C1 C1(C(=O)NCC2CCN(C(Cc3cnc(C)[nH]3)=O)C2)CCN(C)C1C C1(N(C(Cc2scc(CC)n2)=O)C)CCCCN(C(C2CCC(C)(C)OC2)=O)C1 CC1CC(C(N2CC(C(N)=O)(CNC(=O)CC3CCN(C)CC3)C2)=O)CC(C)C1 C1(C)(NC(c2ccc(COC)o2)=O)CCCCC1C(=O)NCC(F)F C(N=c1[nH]c(=NCC(=O)N2CCCO2)[nH]c2c1SCC2)c1cc(N(C)C)ncc1 n1(C(C)C)nnc2c(N(CC(C)CNC(C3(C(C)C)CC3)=O)C)ncnc12 N1(CCCNC(c2ccccc2)=O)CCN(c2c(-c3cn(C)nc3)cco2)CC1 c1(C(=O)NC2C(C#N)CN(C(=O)OC(C)(C)C)CC2)cc(=O)c2ccccc2o1 c1(C(N2CC(N(C(C(c3c(C)cccc3)C)=O)C)C2)=O)cc2n(n1)CC(F)C2 N(C(=NCCc1ccnn1C)NCC12CC(CCO1)C2)CC(=C)C C1(NC(c2c(C)nc(N(C)C)s2)=O)CN(C(=O)C2=CCCCC2)CCC1F c1(CNc2c(C(N3C(C(N)=O)CCC3)=O)cc(Cl)nc2)cn2cc(Br)ccc2n1 c1(NC(CCC2(NC(c3c(C)nn[nH]3)=O)CCC2)=O)cncc(Cl)c1 c1(C(N(CC(C)NC(C2CC(C(C)C)C2)=O)CC)=O)cc(C2CC2)on1 C(C(C)(C)N=c1[nH]nc(C(C)(C)C)o1)NC(C=C(C)C(F)F)=O C(=O)(C1CCCc2nc[nH]c21)NC12C(CN(C(C3(CCS(N)(=O)=O)CC3)=O)C1)C2 C1(C(=O)NCC(CC(=O)NC2CCCN(O)C2=O)O)CC2(CCC2=O)C1 C1(CCCCC#N)NC(=O)N(CCNC(C2CCOCC2)=O)C1=O c1(C(N2C(CC(=O)O)CC2)=O)coc(Cn2cc(CC3CC3)nn2)n1 c1(Cc2cn(CCC(=O)NC(C(C)F)C)nn2)cccc(C#N)c1 N1(C(C2(COC)CN(C(=O)CCOCC3CCC3)C2)=O)CCNC(=O)CC1C N1(C(c2cc(OC)no2)=O)CC(C)CN(C(=O)CC2(C)CC2(Cl)Cl)C(C)C1 C1(CCC(=O)OC(C)(C)C)CCC(CN2CCC2C2(OC(C)(C)C)CC2)C1 C1(C(=O)NCCSCC(C)C)CCCCCN1C(C1CCC=CCC1)=O Cc1cccc(CNC(C2(CNC(C3CC(=C4CC4)C3)=O)CC3(CC3)C2)=O)n1 c1(C(=O)NC(C)CCNC(c2cscc2Cl)=O)cnn(C)c1-n1cccc1 c1(C(=O)NCC2CCCN(C(C3CC34CC4)=O)C2)nc(C2CC2)ncc1Cl N1(C(c2c(F)cccc2Cl)=O)CCN(C(C2CCO2)=O)CC2(CC2)C1 C(C)(CCCCNC(C1(n2cccn2)CCC1)=O)NC(C1CCN(CC)C1)=O c1(C(N2C(C(=O)NCCCCN3CCC3)(CC)CCC2)=O)nnc(O)nc1O N1(CC(=O)N(CC(=O)NCCC2(NC(C3CC3)=O)CCC2)C)CCNC(=O)C1 N1(C(C(=O)Nc2c(C)cc(N3CCC3)cc2)=O)CC(CO)OC2(CCCOC2)C1 C1(CNC(c2ccn(C(CC)CC)n2)=O)CCCCN1C(=O)C(C(C)C)SC C1(NC(C(COC)C)=O)CCC2CN(C(=O)Cc3nncs3)CCC2C1 S(=O)(=O)(c1cccnc1)N1C(CC(=O)Nc2ccc(C)cn2)COCC1 C1(CNC(C(C)OCC(C)C)=O)CCN(C(C2CCC=CO2)=O)C1(C)C C1(NC(C2(CCC)CCC2)=O)CCCN(C(C2(C)CC(C)C2)=O)C1 C(=O)(C(C)(CC)C(=O)N(CC(C)(C)CNC(C1CCCN1C(C)C)=O)C)OCC C1(CC)CN(C(c2cnnn2C(C)C)=O)CCC1NC(c1cc[n+]([O-])cc1)=O N1(C(c2cnc(S)nc2)=O)CCC2(CC1)CN(C(C1CCCO1)=O)CC2CO N1(C(C)=O)CCOC(C(=O)NCC(C)NC(c2cc(C(N)=O)c[nH]2)=O)C1 NC(=O)CCC(=O)NCC1CC(O)CN1C(C1C(F)(F)C12CC2)=O N1(C(C2(OC)CCSC2)=O)CCC(C2CCN(C(C3CC(C)(C)C3)=O)CC2)CC1 C1(C)(NC(c2scc(C)c2Cl)=O)CCCN(c2ccc(C(F)(F)F)cn2)C1 Cc1cccc(C(=O)N(C2CN(C(c3ccc(SC(F)(F)F)s3)=O)CC2O)C)c1 c1(-c2cn(C3(C(N4CC(=O)NCCC4)=O)CC(F)(F)C3)nn2)c[nH]c2ncccc12 N1(Cc2n(CC(=O)NCC)nc(C)c2)CCC2(CC1)OCCC2C(=O)OC Cc1cc([N+](=O)[O-])cnc1C(=O)OCc1cnc(C)c(Cl)c1Br c1(-c2cn(Cc3cc(C(=O)NC(CC=C)C)sc3)nn2)cnccc1C(=O)O C(=O)(CC(C)(C)C(C)(F)F)N1CC(C)C(NC(CSC(C)C)=O)C(C)C1 N1(C(C(C(C)O)C)=O)CC2CCC(CNC(c3csc(Cl)c3)=O)C2C1 N1(COCCC(C)n2ccnc2)CCN(c2ccc(OC(F)(F)F)cc2)CC1 c1(C(=O)NCC2(NC(C(COC)C)=O)CC2)cccc(S(=O)(=O)N2CCCC2)c1 c1(NC(CCC2(C)CN(C(=O)CO)C2)=O)c(C#N)cnn1-c1ccc(I)cc1 Cc1cn(C)cc1C(N1CCC(C(C)NC(=O)CCCn2ccnc2)CC1)=O C12(NC(=O)NCC3CC(OC)(OC)C3)CCCC1(CO)C2 c1(C(=O)NCCCCn2cc(CCCC)nn2)cc(S(C)(=O)=O)cnc1O C1(NC(C(C(C)O)N(C)C)=O)CC2CC1N(C(=O)CSC(C)(C)C)C2 C1(C#N)(C(=O)NCC2CCN(C(c3c(C)ccnn3)=O)CC2C)CCN(C)CC1 N1(C(CCC(=C)Br)=O)CCC2CCC(C1)N2C(=O)COCCCC(C)C N1(C(c2ccc(NC(=O)NC(C(=O)OCC)C)cc2)=O)CCC(C)(COC)CC1 N1(C(C(C)Cc2ccccc2)=O)CC2(NC(c3cn(C)cn3)=O)CC1C2 C1(C#N)(C(N2CC(n3cc(C4C(C(=O)OC)C4)nn3)C2)=O)CCCC1 C1(Cn2cc(C3CC(OC)(OC)C3)nn2)CCN(C(=O)C(C)Br)C12CC2 C1(NC(c2c(CC)cco2)=O)C2CC3C1C3C2C(N1CCC(F)CC1)=O CCC(CC(=O)NCCC1CCN(c2nnc(CC(F)(F)F)s2)C1)C1CCC1 C1(=CCNC(C(C)(C)NS(C)(=O)=O)=O)CCN(C(=O)CC2(O)CCC2)CC1 c1(C(N2C(C(C)NC(C3CC=CCC3)=O)CCC2)=O)ncc([N+](=O)[O-])n1C C(CC(C)(C)CC(=O)N(CC(=O)NCCSCCCO)C1CCC1)OC c1(N2CCCN(C)CC2)nc2ccc(Cl)cc2c(=NCCc2nc(=N)[nH][nH]2)[nH]1 C(=O)(C(C(C)c1ccccc1)NC(C)CN1CCC1)OC C(CC)(CCCC(=O)N1CCC(C2(C)CC2)C1)NC(C(C)(C)OCCC)=O C1(CCC)CN(C(=O)C(c2scnc2C)C)CCN1C(=O)CN(CC)CC C(CCC(C)(C)NC(=O)CC(C)CF)NC(C=CSC)=O C1(CNC(CN(CCC)C)=O)CCN(C(=O)CC2(O)CCOC2)C12CC2 C1(CC)CC(C)CN1C(=O)C=CCNC(C1(CC)CCOC1)=O C(=O)(C(C)CC(=O)NC1CCCCC1NC(c1c(Cl)n[nH]c1C1CC1)=O)OC c1(C(N(CCOCCCN(C(=O)C=CBr)C)C)=O)nncs1 N1(C(C2CC(C)(CC)C2)=O)CCCC(CC)C1C(=O)NC1CC(F)(F)C1(C)C C(=O)(CN=c1[nH]c(N2CCC(n3cccn3)C2)nc2c1CCCCC2)N(C)CC C(CC(C)(C)CC(=O)N1CCC(NC(c2cc(CC(C)C)[nH]n2)=O)C1)OC C12(C(=O)OCC)CC(NC(c3ncoc3C)=O)(C1)C1(CCC1)O2 C(=O)(CCCC(=O)N(C)C)N(CCC(=O)N(CC(O)C1CCC1)C)CC=C N1(C(Cc2nc(C(C)C)sc2)=O)CCCC(N(C(=O)Cc2c[nH]ccc2=O)C)C1 C1(CCNC(=O)C=Cc2ccncc2)CN(C(C2CC3(CC3)C2)=O)CCS1(=O)=O c1(C(=O)NC2C(NC(Cn3ncc(C#N)c3)=O)C2)cc2ccnc(Cl)c2[nH]1 c1(CN(CC(c2c(C)ccc(C)c2)O)C)c(C)c(C)cc(C)c1C Cc1nc[nH]c1C(=O)NC12CC(NC(C3CSCN3C(=O)OC(C)(C)C)=O)(C1)C2 Cc1cc(C(N2CC(c3noc(C(C)C)n3)C2)C)c(C)[nH]1 C(CC(O)C(=O)NCc1cc(C(N)=O)co1)NC(C(C)(O)C1CCC1)=O CC1Oc2ccc(CN3CCCC3CCCc3ccccc3)cc2NC1=O C1(C(=O)NCC2(O)CN(C(C(C)OCC(C)C)=O)C2)OCCN(C)C1=O N1(C(C(C)=C(CC)C)=O)CC(NC(=O)CP(C)(C)=O)C2(CC2)C1 C1(C(=O)NC(c2cn(Cc3nc(C(=O)O)cs3)nn2)C)CCC2(CC2)C1 C1(NC(CN(CCC)C)=O)CCS(=O)(=O)C12CN(C(C1(C)CCC3CC3C1)=O)C2 C(=O)(C(C)(C)CS(N)(=O)=O)NC1CCN(C(c2n[nH]c(C)c2F)=O)CC1 C(CN=c1cc[nH]cc1S(=O)(=O)NCC1CCCCCOCC1)N(C)C Cc1[nH]nc2ncc(C(=O)NC3CN(C(c4ccccn4)=O)CC(C)(C)C3)cc12 c1(CC(N2CCC(NC(c3cc(CC)nnc3C)=O)C2)=O)nc(F)c(F)cc1F N1(C(C(CCC)CNC(=O)C(CN(C)C)C(C)C)=O)CCc2cccc(O)c21 N1(C(COCC(=O)NC)=O)CC(C)(C)CCC1CNC(c1cc(C)nc(O)c1)=O CON1CCC(CC(=O)NC2CCCC2NC(c2cc(Cl)ns2)=O)CC1 C12(C(=O)NCC(C)NC(C3CCN(C)C(=O)C3)=O)CCCN(CC1)S2(=O)=O CCC(CCC(=O)N1CCCC(NC(c2oc(SC)cc2C)=O)C1)OC C(=O)(C1c2ccccc2C2CC1C2)NCCCN(C(c1c(C)nco1)=O)C C1(NC(C2CC(C)(C)CN(C(N)=O)C2)=O)CCN(C(=O)C(C(C)(C)C)N(C)C)O1 n1(CC)cc(CN2C3CCC2CC(NC(=O)C=CC(C)C)C3)c2cccnc12 N1(C(C2CCCC(C)C2)=O)CCCC(C)(C)C1CNC(=O)CCC1CCC(C)O1 N1(C(C2(CC)CC=CC2)=O)CC2COCCC2(NC(=O)C(=O)NCC(F)(F)F)C1 c1(NC(C(C2CCN(C(C3CCCCC3)=O)C2)C)=O)cnc2c(c1)CCC2 c1(C(=O)NC2CCCC(NC(C3N(C)CCCC3)=O)C2)coc2c1COC2 C1(CN(CC(=O)OC)CC)CCN(C(=O)CNc2ccc(Cl)cn2)C(C)C1 CCCC(CC)CCC(=O)NC1CC2CCC(C1)N2C(c1cnc(C)n1C)=O C(=O)(CC(C(F)(F)F)NCc1cnc2ccccn12)N1CC(=O)OCC1C(=O)O c1(C(C)C)nccn1CC(=O)NCC(C)N(C)C(C1CC1)=O.C(C)C CCS(=O)(=O)CC(C)N(C)Cc1sccc1OC c1(C(=O)NCC2CN(C(=O)C=Cc3cscn3)C2)cc(Cl)cnc1O C(=O)(CC1COc2ccccc21)NCCCCN(C(=O)C1=NOC2(CCC2)C1)C C1(C)(C(N(CC(C)(C)NC(c2c(C)nccn2)=O)C)=O)CCc2ccccc2C1 c1(NC(c2c(CNC(=O)CSc3cn[nH]c3)cc[nH]2)=O)cc[nH]c2nccc1-2 N1(C(CC2CC(OC)C2)=O)CCCC1CNC(=O)Cc1csnc1C C1(C(=O)NCCCOCCN(C(CC(C)N(C)C)=O)C)CCCCN1S(N)(=O)=O CCC(C)(C(=O)NC(C)CN(C)C(C1CCN(C(C)=O)C1)=O)OC C1(C(=O)NCc2scc(C#N)n2)C2CC3C(C2NC(c2nnsc2N)=O)C13 CCC(O)C(F)(F)C(=O)NC1CC(CNC(=O)CSCc2cccc(C)c2)C1 c1(C(CC)C)ccc(C#N)c(C(=O)OC)n1.C12CCC(CC1)C(=O)NC1C(C1)N2 c1(C(N(CCC)CCNC(=O)CC2CCCC2(F)F)=O)ccc2nc(O)[nH]c2n1 c1(CNC(C2(C)CCCO2)c2nnnn2CC2CCOCC2)ccc(F)cc1Br C1(CC=C)(C(=O)NCC2CCNC(=O)C2)CCN(C(=O)Cn2cc(C)cn2)C1 C(=O)(C1=CCCSC1)NC(C)C(c1ccccc1)NC(c1cc(O)nn1C)=O C1(C(=O)NCC(CNC(C2(CC)CC2(F)F)=O)(C)OC)CN(C)C(=O)N1 N1(C(C(N2CC(OC)CC(OC)C2)=O)=O)CCCc2cc(Br)ccc2C1 N1(C(c2[nH]cc(C)c2)=O)CCCC(C2CC2NC(c2cc(C)cc(Cl)c2)=O)C1 CCC(COC)(CC)C(=O)NC(C)CC(=O)NCCC(O)CO c1(C(N2CC(CNC(C=C(C)C3CC3)=O)N(C)CC2)=O)cnc2ncnn2c1N C(=O)(CC(C)CC(=O)OC1CC(F)(NC(=O)OCCOCC)C1n1cccn1)OCC C1(NC(C(C2CCCCC2)C)=O)CCC(C)(NC(C2CCC3CC23)=O)CC1 C(=O)(C(C)(O)CCN(C)C)N1C(CO)CC(NC(C2(COC)CC=CC2)=O)C1 c1(OC)cc(F)c(C(=O)NCCCC(C)NC(c2ccc(O)nc2)=O)cc1OC c1(NC)cnccc1C(=O)NCC1(CCNC(C2(CC(C)C)CC2)=O)CC1 Cc1oc(C#N)cc1C(N1CCCC(NC(C2(CO)CC2(F)F)=O)CC1)=O C=C(C)C1CN(C(=O)CC2(NC(=O)CC3C=CCCC3)CC2)CCO1 n1(CC)ncc(C(=O)N(CCNC(C2CCCCN2C(N)=O)=O)C(C)C)c1C C1(C(N2CCC(CNC(C3CC(C(C)C)C3)=O)C2)=O)(CC)CCCCC1 CC1(CNC(=O)CC2COCCOC2)CCN(C(C23CC4CC2C3C4)=O)C1 C(=O)(CC(F)(F)C(F)F)NC1CCN(C(C(C)CN2CCOCC2)=O)CC1F c1(C(=O)Nc2scc(C(=O)Nc3ccncn3)n2)c(O)c(Cl)cc(Cl)c1Cl C(CN=c1cc[nH]c(=NCCc2ccc(C(F)(F)F)cc2)[nH]1)(C(C)(C)C)N(C)C CN1CC=CCC1CC(=O)NCC1(NC(=O)Cc2cncc(F)c2)CCOC1 Cc1nc(C(F)(F)F)oc1C(=O)NC1CC2(C1)CC2NC(=O)CC1CC1(Cl)Cl N1(C(c2cc(Br)no2)C(=O)NC2(C)CC2)CC2CCC(CC2)C1 C=CCCCCC(C(=O)NCCCC)N1CCCC(Cc2nccn2C)C1 Cc1nc2sccn2c1C(=O)NC1CN(C(=O)CC2(O)CCCC2)CCC1CO n1(C(C)C)cnc(C(=O)NCCCCCN(C)C(C2CCCC2O)=O)c1 C1(NC(C2N(CCC)CCC2)=O)CN(C(=O)CN2C(=O)CCC2=O)CC12CCC2 CC(C(=O)NC1CC12CCN(C(C1CCCN1N=O)=O)C2)S(N)(=O)=O c1(N(CC)CC)ccccc1C=CC(=O)NC1CC(N2CC3CCC2C3)C1 c1(C(=O)NC(C)CCNC(=O)C(C)(C)C(F)F)cnc2c(n1)CCCC2 C1(NC(C(=O)Nc2ccc(OCCCOC)cc2)=O)CCCC2(CC1)CC2 c1(C(N2C(CNC(c3cncc(N(C)C)c3)=O)CC2)=O)scc2c1OCCO2 C1(NC(c2ncn(CC)c2)=O)CCCC(NC(C2(C(C)(C)C)CCCCC2)=O)C1 c1(CCNC(=O)Cn2cncn2)ccc(-n2cc(CC3(O)CCC3)nn2)cc1 c1(C(N2CCOC(C)C2C(=O)NC2C3CCCCCC23)=O)cccc2cncn12 Cc1c(C(=O)NCCN(C(C2(C(C)C)CCC2)=O)C2CC2)noc1C1CC1 Cc1nc2ncccc2cc1CC(=O)NC(C)CNC(C1CC2C=CC1C2)=O C1(CNC(=O)CC2CCCCO2)CCCCN1C(C1CCCCCC1)=O N1(C(C(C)(C)C2CC2)=O)CCCCC(NC(C2(c3ccccc3)CC2(Cl)Cl)=O)C1 c1(C(=O)NC2CC(NC(C(C(C)C)(C)C)=O)C2)cc(Br)c2[nH]cnc2c1 N1(C(c2cocn2)=O)CCCC2(CCCN2C(=O)C2CCCc3ccnn32)C1 C(=O)(CCCCCC#N)NCC1=NOC2CCCC12.CC1(C)C2CC1CC(=O)N2 Cc1c(CC(N2CCN(C(C3CC=CCC3C(F)(F)F)=O)CC2)=O)ncn1C C1(C(=O)NC(C2(O)CCCC2)C)COC2(C1)CN(C(=O)Cc1ccnn1C)C2 N1(C(c2c(C#C)c[nH]n2)=O)CC(O)CC1(C)C(N1CC2(CCOC2)C1)=O c1(C(N2CCC(NC(c3ccc(Br)c(C)c3F)=O)C2)=O)cccc2ccncc12 c1(NC2CC(NC(=O)C=Cc3cocn3)C23CCC3)nc(O)c2ccccc2n1 N1(CC)C(=O)CC(C(=O)N(C2CCOCC2)CC(=O)NC)C1c1cccnc1 C(C(C)N=c1[nH]n(C)c(=O)n1C)c1ccc(C)o1 Cc1c(C(=O)N(C(C)CN(C(=O)COC2CC2(F)F)C)C)cnc2ccnn12 c1(C(=O)NCC2N(C(C3CC(C)C3)=O)CCCC2(C)C)ccc2ccccc2n1 N1(C2CN(C(C)C(C)CC(=O)OC(C)(C)Cl)C2)CCN(c2ccccc2)CC1 N1(C(c2oc(C)c(CO)c2)=O)CC2(CC(NC(=O)CCOC3CCCOC3)C2)C1 c1(C2(NC(C)CC3CCN(C(=O)OC(C)(C)C)C3)CCC2)ccc(Cl)cc1 C(=O)(CCC(=O)NN(C)C)NC1(CCCCNC(C2C(C)SCCC2)=O)CC1 c1(SC)ccc2cc(C(=O)NC34CC3CN(C(c3cccc(C)c3)=O)C4)[nH]c2c1 N1(C(C2N(CC(C)C)CCC2)=O)CCCC(C)(CNC(c2ccccc2O)=O)C1 CCCC(C(=O)N(CCCNC(=O)C(=Cc1cnn(C)c1)C)C1CC1)NC(N)=O C1(C(=O)NCCCN(C(=O)CCCNS(C)(=O)=O)C)CCCN(C(=O)C2CC2)C1 c1(C(=O)NC2(CC(=O)NC3CC(=C)C3)CCC2)c[nH]nc1C C1(C)(C(=O)NCC2(C)CCN(C(CCC3CC(OC)C3)=O)C2)CCC(F)(F)C1 c1(C(=O)NC2CCC(NC(c3n(C)ccn3)=O)C2)ccc(Br)c(Cl)c1F C1(CNC(CC(=O)OC)=O)CC(C(=O)NC(c2ccc(C)cc2)C)=NO1 N1(C(CC(C)F)=O)CCCCC1C1(CNC(=O)COC2(C)CCC2)CCOCC1 c1(OCC)ccccc1CCC(=O)N(CCNC(C1(F)CC=CCC1)=O)C1CC1 c1(C(N(C(CNC(C2CC(C)(c3ccccc3)C2)=O)C2CC2)C)=O)cc(O)ncn1 N1(C(C2C(NC(C3(OC)CCCOC3)=O)CCC2)=O)CCC12CC(O)C2 CC1(C)CCN(C(=O)C=Cc2cc(Br)cs2)C1c1ccccc1 C1(NC(C(COC)(C)C)=O)CC2CC1CN(C(=O)C1=CCCC1)C2 c1(CC(=O)NC2(C)CCN(C(C3CCCO3)=O)C2)ccc(S(N)(=O)=O)s1 CCCC(C(O)C(=O)NC1(C)CC2(CC2)C1)NC(C1CC(C)(C)CO1)=O C12(C=O)C3C4C1C1C2C3C41C(=O)OC.c1(C(N(CC(C)O)CCN)=O)c[nH]nc1C CCCCCC(F)C(=O)NCC1CN(C)CCN1C(C1CCS1(=O)=O)=O C(=O)(CS(=O)(=O)CCO)N1C(C)CC(NC(C23CC(F)(C2)C3)=O)CC1 c1(OC)cc(C)c(C(=O)NCC(CNC(=O)COCCCF)OC)cn1 C1(C2CCN(c3ncc(Cl)cn3)C2)(NC(C2CCCCC2O)=O)CC1 c1(-c2cn(C3CCC(C(=O)NC(C)C(=O)NCCO)C3)nn2)cccc(CO)c1 C(C(C)C(F)C(=O)NCc1ncc(CC)[nH]1)NC(c1n(CC#C)ccc1)=O N1(C(C2Cc3ccccc3C2)=O)CCOCC2(COCCN2c2nncs2)C1 c1(OCC(N2CC(C(=O)NCC3CC(C)(C)C3)OCC2)=O)ccccc1[N+](=O)[O-] c1(C(=O)NC2CCC(C(=O)NC(C3CCC3)C)C2)cccc(-c2ccoc2)c1 Cc1cc(NC2CS(=O)(=O)CC2C)ncc1S(=O)(=O)N1CCC(CCOC)CC1 C(=O)(CCC(C)S(C)(=O)=O)NC1(CC=C)CCN(C(=O)CCS(C)(=O)=O)C1 c1(C(=O)NC2(C(N(CCCCCC=C)C)=O)CC(F)(F)C2)cccn2nccc12 c1(C(N(CCCNC(c2nc(CC)sc2)=O)C(C)C)=O)ccc(=O)n(CCF)n1 C=CC(CC)C(=O)NC(c1nc(=O)o[nH]1)C N1(C(C#CC(C)(C)O)=O)CCCC2(CNC(=O)CS(N)(=O)=O)CCCC12 C12(NC(C3CC(C#N)(O)C3)=O)CCC(C1)N(C(=O)CC1(O)CCCCCC1)C2 C1(NC(c2ccc(COC)[nH]2)=O)CCN(C(c2ccoc2C(F)(F)F)=O)CC1O c1(CCC)cc(C(=O)NC2CCN(C(c3cn(C)nn3)=O)C2C)sc1C CC(CC(=O)N1CCN(CC2CN(C(=O)OC(C)(C)C)C2)CC1)C(F)(F)F CC(CC=CCl)(C(=O)NCC1(NC(C2CCC(=O)C2)=O)CCC1)c1ccccc1 C(c1ccc(F)c(F)c1)=C(C)C(=O)NCC(CO)NC(=O)C(C)C(O)C(C)C CC1CCC(N=c2[nH]c(=NCc3cccc(C(C)(F)F)c3)[nH]c3c2COC3)CC1 Cc1ccc(C(=O)NC2CC3CC(NC(C4CCCS4)=O)C2C3)c(C2CC2)c1 c1(CNC(C2C(NC(C(C)OC)=O)COC2)=O)ccc(=O)n(C)c1 c1(CNC(C(C)=C(C)C)=O)nc2c(s1)CCN(C(C1CCS(=O)(=O)C(C)C1)=O)C2 CC(C(F)C(=O)NCCOCCNC(c1cn2cc[nH]c(=O)c2n1)=O)C(F)(F)F Cc1cc(C(=O)NCC=CCNC(=O)C(C2CCCO2)C2CC2)cs1 C12C3CN(CC13)N(C(C)C)CCNC(=O)C2.c1(C(=O)OC(C)(C)C)ccoc1 C(CC(C)(C)CNC(=O)CNC=O)NC(c1cn(C(C)C)nc1)=O N1(C(CNC(c2ccon2)=O)=O)CC2(CC(NC(=O)CC(C)n3cccn3)C2)C1 N(C(C(=O)N(C)CCNC(=O)C(F)C1CCOC1)=Cc1cccs1)C(C)=O N1(C(CCSCCC)=O)CC=C(CC(=O)NCc2coc(C)n2)CC1 C#CC1CCN(C(C2CCC(NC(=O)CCCCN(C)C)C2)=O)C1 CN1C(=O)CCC1CC(=O)NCC1CC1NC(=O)CCCc1cnn[nH]1 C1(C(N2CC(F)(C(=O)NCCC(C)N3CCC3)C2)=O)CC(C)N(C)C1 CN(C[Si](C)(C)C)C(=O)C(Cn1cncn1)NC(=O)CCc1cnoc1 Cn1ccc(=NCC(C)(CC(=O)O)NC2CN(C(=O)OC(C)(C)C)C2)[nH]1 N1(C(CCSC)=O)CC(Nc2ncnc3[nH]cc(C(N)=O)c23)C2(CCOCC2)C1 C(CN=c1nc2c(Br)csc2c[nH]1)(N(C)C(C1CCS(=O)(=O)CC1)=O)C1CC1 Cc1ccc(C(=O)NC(C2CCN(C(=O)CSCc3ccc(Cl)s3)C2)C)nc1 C12(NC(CC(CC)C3CC3)=O)CC(C)(C1)OC21CN(C(=O)C(O)C2CC2)C1 c1(NC(CONC(C2(C)CC(C)OCC2)=O)=O)ccc(N=[N+]=[N-])cc1 N1(C(C2C(C(C)O)C2)=O)CC(CNC(=O)C(C)(C)C2CCCCC2)OC(C)(C)C1 n1(C(N(C2CCN(C(C3(C#C)CC3)=O)C2)C)=O)cc([N+](=O)[O-])nc1C C(=O)(C(N)CC1CC1(F)F)N(CCCC)C(c1ccccc1)C C(C(C)CNC(=O)CC1CC(NC(=O)CC2CCOC2)C1)OC CCC(C)C(O)CC(=O)N1CC(O)(C(F)C(=O)Nc2c(C)csc2C)C1 c1(C(=O)NC(C2CCOC2)CNC(C2=C(C)OCC2)=O)cc2c(nn1)CCC2 C1(CCNC(C2(C(=O)OC)C(=C)CC2)=O)CCCN(C(c2nn(C)cc2N)=O)C1 c1(CC(N2CCN(C(c3cc4sc(Cl)cc4[nH]3)=O)CC2)=O)cn2c(n1)CCCC2 O=C(C1CC=Cc2ccccc21)NC1CC2(C1)CN(C(c1ccc[n+]([O-])c1)=O)C2 c1(CCC(=O)NC2CCC(C)(NC(CSC)=O)CC2)ccccc1N=[N+]=[N-] c1(N(C2CN(C(Cc3c(COC)cccc3)=O)C2)C)ccc(C#N)nn1 C1(N(C)C(C2(C)CC2Br)=O)C2CC1N(C(=O)CN1CCC(O)CC1)C2 c1(C(N2C(CNC(C3C(OCC)C3C)=O)C(C)CC2)=O)cc(F)cc(OC)c1N C(C)(N=c1ccnc(Cl)[nH]1)C1CCN(C(CCC(=C)Br)=O)CC1 N#CC1(NC(c2cccc(C3CCC3)c2)=O)CCN(c2ncc(Br)cn2)C1 CC1(NC(c2cc(C3CC3)nc(O)c2)=O)CCCN(C(C2CC3CC2CO3)=O)C1 C(C(N=c1[nH]ncs1)C1CCC1)NC(=O)C=Cc1cccnc1 N1(C(CCC(=O)OC)=O)CCOCC(C)(CNC(C2COCCC2(F)F)=O)C1 N1(C(c2[nH]cc(CC)n2)=O)CC2CC1CN(C(c1ccc3c[nH]nc3c1)=O)C2 Cc1nn(C)c(C)c1C(=O)C(N1CCC(NC(=O)CSc2nccn2C)CC1)=O C12CN(CC1O)C2=O.c1(NC(=O)CSC(F)(F)F)cccc(-n2cnnn2)c1 CC1(C)CC(C)(CNC(=O)CC2CN3CCC2CC3)CN1C(=O)Cc1ccon1 c1(NC(CC(CN(C)C(C2C=CCC2)=O)O)=O)ccc(C2CC2)s1 CC1CCCC(C)N1CCC(=O)NCC(C)CNC(C1(C2CCCO2)CCC1)=O c1(C(=O)NC(C)CCNC(C2(Br)CC2(C)C)=O)ccnnc1O c1(N(CCC)C)cccc(-c2nc(-c3cc[nH]n3)nn2CCF)c1 c1(C(=O)NCC=C)nc(C(=O)NCC(CO)NC(=O)C(c2ccc(Cl)s2)=O)cs1 c1(CN(C2C(=C)CC2)C(=O)NCC2CCCCC2)cc2ccc(F)cc2s1 C(=O)(C(CC)C(F)(F)F)N(CCC)CCNC(=O)C(c1nc(F)ccc1Cl)C C12(CNC(c3cc(C)n(C)n3)=O)CCCC1CCN2C(=O)CC=C(Cl)Cl C1(CNC(c2cccc(C)n2)=O)CN(C(c2ccn(C)c2C2CCC2)=O)CCCO1 CCC(CNC(c1cc(C)c[nH]1)=O)(CC)NC(=O)C(C)Sc1ccccc1Cl c1(C(=O)NCC=CCNC(c2n[nH]cc2Cl)=O)cnnn1-c1ccccc1 CCC(CC)(CCOC)C(=O)N1CC(CNC(=O)CCCC(F)(F)F)CC(C)C1 c1(C(N(CCC(C)NC(C2(C#C)CCC2)=O)C)=O)n[nH]c2ccc(F)cc12 C(C)(CCCO)(c1n(C(CC)C)nnn1)NC(c1sccc1Cl)C N1(C(c2cc(C)sc2N)=O)CCC2(CCN(C(c3csc(C4CC4)n3)=O)C2)C1 c1(CNC(NCC2CNC(=O)O2)=NCC2CCC2)ccc(Br)cc1Cl N1(C(C2(CC)CC2(F)F)=O)CC2CCN(C(=O)Cc3nonc3C)CCC2C1 c1(OC)cc2ccccc2cc1C(C(=O)NC1CCCCC1)N(CCCO)CC C1(OCC)CCC(C(=O)N(CCCN(C)C(c2ncn(C(C)(C)C)n2)=O)C)CC1 c1(C(=O)NCCOC2CN(C(C(C(C)O)N(C)C)=O)C2)n[nH]c2c1COCC2.C(N)(=O)N N(C1COCc2cc(Br)ccc21)C1C(F)(F)CCC1 c1(C(N2CCCC(n3cc(CCNC(=O)OC)nn3)C2)=O)cc(C)cc(Br)c1 Cc1ccc(C(N2CC3(CC3)CC2C(=O)NC2CC(CO)C3CC23)=O)nc1C n1(CC(=O)NCC(C)N(C(c2onc(C)n2)=O)C)c(C)ccc1C C(C(C)C(=O)NOCCC(C)C)N(C(c1cc(CC)ncc1)=O)C C1(O)(CN(C(COC(CC)C)=O)C)CCN(C(c2cc(C3CC3)n(C)n2)=O)CC1 c1(CC)nc(O)c(C(=O)N(C(C)CN(C(=O)Cc2ccc(O)cc2)C)C)cc1C c1(C(N(C2CCCC(NC(=O)CN(C)CCO)C2)C)=O)cccc2oc(=N)[nH]c12 C(=O)(C1CCSc2ccccc21)N1CC2=C(CN(C(C(C(C)C)SC)=O)C2)C1 N1(C(CCC(C)OCC)=O)CCC2CN(C(=O)C(C)=CCO)C2C1 C(=O)(CC(C)C(=O)NCC1(NC(c2coc(C3CCCCC3)n2)=O)CCC1)OC c1(OC)ccc(CC(N2CCC(N(C(=O)COC3CCCC3)C)CC2)=O)cn1 N1(C(C2C(OC)C(O)C2)=O)CCc2sc(-c3cn(-c4nccs4)nn3)cc2C1 N1(C(CC2C(NC(C=Cc3cn(C)nc3)=O)CC2O)=O)CCOCCC1C(N)=O C(=O)(C(O)C(C)(C)C)NCC(CC)NC(c1ccc(Br)cc1)=O c1(C(N2CCCC(N(C(=O)CC3CC3)CC)C2)=O)c(C)cc(Cl)cc1C c1(C(N(C2CN(C(c3cn(C)nc3Cl)=O)C2)C)=O)ccc(-c2ccco2)cc1F c1(C(=O)NC2CC(C)(CNC(c3cnc(OCC)s3)=O)C2)cc(F)c(N)cc1F C(=O)(C1=CC(O)C(O)C(O)C1)N1C(C#N)C2CC2C1.C12CCN1C2=O c1(CNC(c2cn(CC3CNCCO3)nn2)=O)ccc2c[nH]nc2c1 N1(C(CCc2ccc(OC(C)C)cc2)=O)CC(C)Sc2ccccc21 CCCCCCCCCC(C(=O)Nc1ccccc1)N1CCc2[nH]nc(O)c2C1 C1(C(=O)NC2C(CNC(Cc3cccc(C)c3)=O)CC2)CC(=O)OC1(C)C c1(OCCC=C)cccc(OC(C)C(=O)OCC(O)CN=[N+]=[N-])c1 c1(OC)ccc(C)cc1C=CC(=O)NCC12CCCC1CCN2C(=O)CN(C)C C1(C)(CN(C(CC2(COC)CC2)=O)C)CCCC1.C1(C2CCOC2)C(=O)N1 C1(C(=O)OC)CN(C(=O)C=Cc2ccc(Br)s2)CC(C)O1 c1(C(=O)NC2CCC(NC(C3(COC)CCC3)=O)C2)cn2c(n1)CCC2 c1(-c2cn(CCC(C)(C)NC(C3N(CC)CC3)=O)nn2)cccc(C(F)(F)F)c1 N1(C(C(=O)NC(C)C)=O)CCC(NC(c2cnc3sccc3c2)=O)C(C)(C)C1 C=CC(CCC)CC(=O)NC(CC(C)CC)C(=O)Nc1ccc(Cl)cc1 CCCCC(CNC(c1nnc(S)n1C)=O)NC(=O)COC1CC(F)(F)C1 c1(COC)cc(=NCC2CCN(C(C3(COC)CC3)=O)CC2C)[nH]c(C(C)C)n1 C1(C2(O)CCOC2)(C(N2CCC(C(C)NC(CC)=O)C2)=O)CC1 C1(NC(C(C(C)C)O)=O)CN(C(c2cccc3cccnc23)=O)CCC12CCC2 Cc1ccc(OCCC(=O)NC2CC3(C2)CC3NC(c2cccnn2)=O)cc1C C1(CNC(c2cc(C)n(C)n2)=O)CN(C(C2CCCOCC2)=O)C(C)(C)C1 C(=O)(C(CCC(C)C)NC(=O)CC1C=CCC1)NCC(C(=O)OC)(C)O c1(OC)ccc(CNC(=O)C(O)CC[S+](C)C)cc1[N+](=O)[O-].C1C(=O)N1 N1(C(=O)C2=CC3(CCOC3)C2)CCOC2(CCN(C(C3CCC3)=O)CC2)C1 c1(C(=O)NC2CCN(CC(COC)O)CC2)cc2cc(F)ccc2cn1 C1(CNC(CCOCCOC)=O)CCC(C)N(C(=O)Cc2nccn2C)C1 N1(C(c2cccnn2)=O)CC2CC(NC3CC(OC(F)F)CN3)CC2C1 C1(C(N2CCN(C3CN(C(C(C(CC)O)C)=O)C3)CC2)=O)CCC2(CCC2)CO1 c1(C(N2CC(NC(C3C(C)CCCC3)=O)C3(C2)CC3)=O)c(F)cc(N)cc1F C1(NS(CC)(=O)=O)CN(Cc2cccc(O)c2)CC12CC2 c1(C(C)(O)C(=O)NC2CCC(NC(C3(F)CCC3)=O)CC2)ccc(F)cc1F c1(NC(C2C3(CN(Cc4cnc(OC)nc4)C3)C2)=O)ccc2ccc(Br)cc2c1 n1(CCCCOC)c(N2CCCC2CN(C)C)nnc1C1CCCCN1C C(=O)(C(N)CCC(=O)c1ccccc1)OC.N1(CC=O)CCN(C=O)CC1 n1(CC(=O)NC2CCC(N3CCCCC3)CC2)cnc2sccc2c1=O n1(CC)nc(C(=O)NCC(C)N(CC(=O)N(C)Cc2nccs2)C)cc1O c1(C(=O)NC2CCCCN(C(CC=CCC)=O)CC2)n[nH]c2ccc(Cl)cc12 c1(NC(=O)NCCN(C(=O)CCC2COC(C)(C)O2)C)cc2ccccc2nc1O C1(C(N2CCC(C(C)NC(=O)CN=S(C)(C)=O)C2)=O)CCOC2(CCCCC2)C1 c1(C(=O)OC)cc2c(NCC(C)N(C)C(C34CC3COC4(C)C)=O)[nH]cnc-2n1 C1(CC)C(NC(c2cc(C3CC3)[nH]n2)=O)CCCN1C(C1CCC(C)(CC)O1)=O N1(C(Cn2ccc(C)c2)=O)CCC(C)C1C(=O)NC1CC1CN(C)C N1(C(C2(CCCC)CCCC2)=O)CCCN(C(c2cncnc2)=O)C(C)C1 C(C)(C(=O)NN(Cc1ccccc1)c1ccccc1)c1cccc(OC)c1 C1(CC)CCCC(NC(=O)CN(CCOC)C(C2CN(C(C)C)C2)=O)C1 N1(C(C(Cc2cc[nH]n2)NC(C(C)CC#N)=O)=O)CC2CCC(C1)C2C#N c1(N(CCCCC=C)C)cc(C)c(S(=O)(=O)N2CCCC2CC(C)(C)C)cn1 CN1CCc2cc(CC(=O)NCC3(C)CCCN3C(=O)CC3CC=CC3)ccc21 C(=O)(CCCCC(F)(F)F)NCC(CC(C)C)NC(c1ccccc1C(C)O)=O c1(CC)nncn1NC(=O)CC(C)NC(C1CCN1C(C)(C)C)=O C1(NC(C2N(N=O)CCC2)=O)CCS(=O)(=O)C12CN(C(C1CC13CC(O)C3)=O)C2 CCCC(CC(C)C)C(=O)N(CCCCN(C)C(c1nc(C(C)C)oc1C)=O)C C1(C(=O)NC2CCC(C(F)(F)F)C2)CCN(C(=O)CCCCC2CC2)CCO1 C(=O)(C(C)c1ccsc1)NCC1(CN(C(C2C(C(=O)OC)C2)=O)C)CC1 C1(S(N)(=O)=O)(C(N2CC(OC)C(NC(c3occc3C(C)C)=O)C2)=O)CCC1 C12(C(=O)OC)CC3CC1C2C3C(=O)Nc1sc(I)cc1OCc1ccccc1 C(=O)(CC(C(F)F)n1ccnc1)NC(C(C)NC(c1n[nH]cc1Cl)=O)(C)C c1(C(N2CCC(N(C(C3C(=C)CC3)=O)CC3CC3)CC2)=O)cc(O)cc(Br)c1 C1(CNC(c2c(C)c(Cl)ccc2)=O)CC2CCC1N(C(C1CCCN1N=O)=O)C2 C(=O)(CCCCC(N)=O)NCC1CCC(NC(c2n(CC)ncn2)=O)CC1 C=CCC(CC=C)C(=O)NC1CCN(C(c2coc(C)c2)=O)C(C2CC2)C1 Cc1ccc(Sc2nnc(C3CCCCC3)o2)cc1F C(=O)(C(CC(C)C)NC(=O)CC1(NC(=O)C=Cc2ccccc2)CCC1)OC C(=O)(C1CSc2ccccc21)NC(CNC(c1c(C(C)C)scn1)=O)CO CC1(C)CN(C(C2CCCN2CC(F)(F)F)=O)CC1NC(=O)CCC1CCOC1 c1(C(=O)NCC(CC)NC(=O)C(C)NC(=O)NC)cccc(C)c1C#N N1(C(c2c(CC)ncs2)=O)CC(CNC(=O)C(c2ccccc2)C)C2(CC2)C1 C1(CC(=O)N(CCCNC(=O)CC(C)O)C(C)C)CCCC1(F)F c1(N(C(C2(NC(C)CCNC(C3CC3(F)Cl)=O)CC2)=O)CCO)ccccc1 c1(C(N(C(C)CNC(=O)C(F)C(F)(F)F)C)=O)cc(Cl)c(Cl)c(Cl)c1 N1(C(c2cc(C)ncc2C)=O)CC23CCCC2(C1)CN(C(=O)Cc1cnns1)C3 C(Cc1ccccc1)(CN=c1[nH]c(N2CCC3(CC2)CC3)nc(=N)[nH]1)OC c1(SC)cc(C(=O)NC2CN(C(=O)CCC3CCCCO3)CC2C)oc1C Cc1cnnc(C)c1C(N1CCC(CCC(=O)NCC2CCCOC2)C1)=O C(=O)(CCCCCCNC(c1cc2n(n1)CCO2)=O)NC1CCC(C(N)=O)CC1 C(CC(C)(C)C)(C(=O)NC(c1ccns1)C)NC(Cn1ncc(C#C)c1)=O C1(NC(=O)C#CC2CC2)CC2(CCN(C(c3ccc(C(F)(F)F)nn3)=O)CC2)C1 N1(C(CC=C=C)=O)CCC(C)C(NC(=O)CCc2ccc(F)c(Br)c2)C1 c1(C(=O)NC(CCC)CNC(c2cc(C3CCC3)no2)=O)c(O)cccc1F N1(C(C(C)(C)N(C)C)=O)CCC2(C1)CN(C(=O)Cc1cn3ccsc3n1)CCO2 Cc1c(C(N2CCN(c3cccc4cnccc34)CC2)=O)oc2ccc(F)cc12 N1(C(Cc2ccc(C)o2)=O)CCCC(NC(=O)CCOC2CC2)C(F)C1 C12(C(=O)NC3CCC(C)(C)C3)CCCC1CN(C(c1cnn(C3CC3)c1)=O)C2 C1(NC(CNC(=O)OCC)=O)CCN(C(C2CCC(F)C2)=O)CCC1CO C(=O)(C(C)CS(C)(=O)=O)N1CCN(C(Cc2cc(C)sc2)=O)CC1CCO N1(C(CNC(C2C(C)C2)=O)=O)CC(C)(C)C(NC(c2ccncc2)=O)C(C)(C)C1 C1(C(C)(C)C)(C(=O)NCC(CC)NC(c2cnn(CC(F)F)n2)=O)CCCCC1 CC(C)(C(=O)NCCNCc1ncoc1C1CCCO1)n1cnnn1 CS(=O)(=O)C1(C(N2CC3CC2C3NC(c2occ3c2CCOC3)=O)=O)CCCC1 c1(-c2ccc(C(=O)NCc3cnc(C)s3)cn2)cc(O)cc(F)c1 c1(C(=O)NC2CCC(CNC(CC(C=C)C)=O)CC2)cnc(C(F)F)cc1C C=C(C)CC(C)C(=O)NC1CN(C(c2csc(-c3cccc(C)n3)n2)=O)CC1OC C(=O)(C1=CCC(C)(C)CC1)N1CC2C(NC(CCCOCC=C)=O)CC(C2)C1 c1(C(=O)NCCC(=O)NCC2N(C(C3C(C)C3)=O)CCCC2)cc(N)nc(Cl)c1 N1(C(Cc2c(C)noc2C)=O)CCN(C(=O)C(C)CNC(N)=O)C2CCC12 c1(C(=O)NCC2C3CN(C(C4(C(=O)OC)C(=C)CC4)=O)CC23)nccn2ccnc12 c1(CC(=O)NC2CC(C)N(C(c3cnc(Cl)c(N)c3)=O)C2)ccc(CO)cc1F c1(CCC(=O)NCC2CCN(C(=O)Cc3ccncc3Cl)C2)cccc(Cl)c1 C1(C(N2CCC(O)(CN(C(=O)C(C)=NOCC#N)C)C2)=O)(CC)CCNC1=O C1(C(N2CC(NC(C)=O)C2)=O)CCC(C(C)C)N1C(=O)Cc1cccc(F)c1 C(CO)(C(=O)N1C(C(=O)N(C2CC=CC2)C)CC1C)OC C1(CC)CC(C)CN(C(=O)C(C)(CO)NC(C2CC(=O)C2)=O)C1 c1(C(=O)NCCC2(O)CN(C(C3CCC(C)C3)=O)C2)ccc2c(c1)OC(C)(C)C2 N1(C(CC2CCN(C(c3ncn(C(C)C)n3)=O)C2)=O)CCC(C2CC2)C1 N1(CCOC)CC(C(=O)NCC2(C)CCN(C(=O)C3=COCCO3)C2)CCC1=O CC1(C)CC(NC(C2CCC(CO)CC2)=O)CN1C(=O)CCCCCF c1(C(=O)NC)cccn2[nH]c(=NC(=O)NCC(C)OC)nc12 C1(NC(c2cnc(N(C)C)s2)=O)CCN(C(=O)COC(F)(F)C(F)(F)F)CC1F CC(C)CC(C(N)=O)NC(C1CCCCN1C(=O)CC1C=NN(C)C1=O)=O N1(C(c2ncn(C)n2)=O)CCCC2(CCN(C(=O)C(C)(F)C(F)(F)F)C2)C1 Cc1cc([N+](=O)[O-])ccc1C(=O)N(C)Cc1ccc(Br)c(Cl)c1 C1(COC)(NC(=O)C(O)C2CC2)CCN(C(c2ccn(-c3cccnc3)n2)=O)C1 C12(C(=O)NC3C(NC(c4c(C)nc(CO)s4)=O)CCC3)CCCC(C)(C1)OC2 N1(C(C(CC)N(CCO)CCN(C)C)=O)CCN(c2ccccc2C)CC1 C1(CN(C(C2CCN(CC)C2)=O)C)CC(F)CN1C(=O)CC(C)(C)SC C1(F)(C(=O)NC2CCN(C(C3C(C)CCC3)=O)CC2F)CCCCC1(F)F c1(C2C(NC(c3ccc(C4CC4C)o3)C)C2)ccc(Cl)cc1Cl n1(CC(=O)NCC2CC(NC(C3CCCN(C(C)C)C3)=O)C2)cnc([N+](=O)[O-])c1 O=C1CCN(CCC2CCC=CCC2)C(=O)N1CCOCC1CCCC1 Cc1c(NCCCN2CCOC2=O)ncnc1NC(c1ccncn1)C c1(C(=O)NC(CCNC(Cc2cc(OC)c(Cl)cc2)=O)C)cccc2oncc12 N1(C(c2c(C)ccnn2)=O)CCCC(NC(c2n[nH]c(C)c2C)=O)C1C C1(C(=O)NC2CCC(COC)C2)CC2(CCN(C(=O)CN=[N+]=[N-])C2)C1 Cc1ccc(C=CC(=O)NCCCN(C(=O)C(C)n2cccn2)C)nc1 c1(C(N2CC3C(NC(CC(C)C4CC4)=O)(C3)C2)=O)ccc(F)c(O)c1 c1(CN(CCS(CC)(=O)=O)C2CC2)cc(=O)oc2c(C)c(O)ccc12 N1(C(C=CCNC(C(CC)(C)COC)=O)=O)CCc2ccncc2C1 c1(C(N2C3CN(C(CSC(C)(C)C)=O)CC2CC3)=O)ccc2n[nH]cc2c1Cl C1(NC(c2ccc(SC)cc2C)=O)C2CCC1CN(C(=O)CN1CCOCC1)C2 Cc1nn(C)cc1CN1CC2C(C(=O)N(CCO)C(C)C)C2C1 c1(OC)ccc(I)c(NCC2CCN(c3nccs3)CC2)c1 Cc1cc(Cl)cc(NC(=O)CC2(C)CN(C(c3ccnc4c3OCO4)=O)C2)c1I c1(C2C(C(N(CC(C)NC(=O)C(C3CCCCC3)=O)C)=O)C2)cccc(F)c1F O=S(=O)(c1cccnc1NCc1cc(C(F)F)no1)NCC1(Cl)CC1(F)F N1(C(C2CC(CCC)C2)=O)CCC(F)(n2cc(CS(=O)(=O)CC)nn2)CC1 Cn1cc2c(n1)CC(C(=O)NCC1(NC(c3cc(C#N)ccc3F)=O)CC1)CC2 N1(C(C2(CC)CCC2)=O)CC2CC1CC2CNC(C1CCC(CN(C)C)O1)=O C=C1C(C(=O)NC(C(=O)NC2CC2c2ccco2)C2CCCC2)C1C(=O)OC C1(n2cccn2)(C(=O)NC(CN(C(=O)Cn2cc(CO)nn2)C)(C)C)CCCC1 C1(c2onc(C)n2)COCCN1C(=O)NC1CCCOC1c1ccc(CO)cc1 C1(NC(CCC2C(C)(C)C2)=O)CN(C(=O)Cc2csc(=N)[nH]2)Cc2nccn2C1 c1(C(N2CCCC(C(C)NC(=O)COC3CC=CC3)C2)=O)cc(CO)cc(Cl)c1 n1(CC)cc(C(=O)NC2(C3CCCN3C(=O)C(C)(C)Br)CC2)cn1 c1(C(=O)NC(CC)CNC(=O)C(CO)NC(N)=O)ccc(O)c(C)c1C CCS(=O)(=O)c1ccccc1C1CC1.N12CC3CC3(C1)CNC(=O)C2=O N1(C(=O)Cn2nnnc2-c2ccsc2)CC2CC(C1)C2NC(CNC1C(C)C1)=O c1(OC)ncc(C(=O)NCC2CNCS2)cn1.C12(CCC1)CC(=O)N2 C1(F)(C(=O)NC(C)(CNC(=O)COC(F)F)C2CCC2)CCOCC1 C1(c2cn(C)nc2)CN(C(=O)CC2CCCCC2)CCN1C(=O)C=CC(C)(C)C c1(-n2c(-c3ccc(C)c(C)c3)nc(CCOC(C)C)n2)cccc2ccccc12 c1(CC(N2CC(C(C)NC(C(C)O)=O)C2)=O)nc(F)c(F)cc1F C(=O)(C(C)(C)C)N(CC(CC)NC(c1coc(C2CCCCC2)n1)=O)C N1(C(C2C(=C)CC2)=O)CC=C(CCNC(c2cncc(-n3ccnc3)n2)=O)CC1 C1(CNC(=O)C2=CCCOC2)CCCC2CN(C(c3ccsc3C(F)F)=O)CC12 C1(NC(C2(CC3CCC3)CC2)=O)CCCCN(C(C2C3COCC23)=O)C1 N1(C(C)=O)CCC(O)C(Nc2ncc(C(=O)O)cc2Cl)C1 C1(C(=O)NCCCCCNC(c2cnc(OC)nc2C)=O)CCc2nc[nH]c2C1 c1(CN(C)CC2CCN(C(C3CC(C)(O)C3)=O)C2)nnc2n1CCCCC2 N1(C(C(CC)O)=O)CC(CNC(c2cnc(C)nc2C)=O)CC1(C)C c1(C(=O)NC2CC(CCNC(COCC(=C)C)=O)C2)cccc(Cl)c1[N+](=O)[O-] C1(C(N(CCC(=O)NC(C(CC)(C)C)C)CCO)=O)CCCCC(=O)C1 Cc1nc(O)ccc1C(=O)NC(CNC(=O)Cn1cc(C#N)cn1)CC(C)C C1(CNC(C2C(C)C2C)=O)CN(C(c2ccccc2C#N)=O)C2(CCC2)C1 c1(OC)ccc(C(=O)NC23CCC(C2)N(C(c2n[nH]c(C)c2Cl)=O)C3)c(F)c1 CCC(CC)C(C)C(=O)NC1CC(NC(c2cc(F)cc(F)c2)=O)C(O)C1 c1(C(=O)NC(CC=C)CNC(=O)CCOCC)cn2ccc(C)cc2n1 CCCCCCC(F)C(=O)N1CCCC1CNC(c1cnnc(C)c1)=O c1(N2CCN(C3CCN(C(CCC(C)SC)=O)CC3)CC2)ccc(C#N)cn1 C1(NC(Cc2c(C)cccc2)=O)CN(C(=O)C=CS(C)(=O)=O)CC(C)(C)C1 c1(OC)c(C(N2CC3CC2CC3NC(c2cc(C)cs2)=O)=O)cccc1F CC1CCN(C(c2sccc2CNC(=O)CCn2ccnn2)=O)CC1O Cc1ccc(CNC2CCC(C(=O)NCCF)OC2)c(Br)n1 C1(C(=O)NCCN(C2CCCCCC2)C(CCCOC(C)C)=O)CC2C=CC1C2 c1(CN2C(C(=O)Nc3c(C(=O)NCCCC)cccc3)CC2)ccc(C)c(O)c1 C1(NC(=O)C(F)=C2CCCC2)CCN(C(c2scnc2C2CC2)=O)CC1CO N1(C(CN(CCC)C)=O)CC(CNC(=O)CC2CC2(Cl)Cl)CCC1C CC(=Cn1ccnn1)C(=O)N1CCC(C)(C)C(NC(C2CCC3CC23)=O)C1 C(=O)(C(C)(COC)CC)N1CCCC(NC(CCSCCCC)=O)C1 c1(C(=O)NC(C#CC)(C)C)nccc2c(Cl)cccc12 c1(C(N(C2CN(C(C3(CO)CCCO3)=O)CC2(C)C)C)=O)ccc2cncn2c1 C1(CCC)(C(N2CCC(O)(CNC(c3ncsc3C)=O)C2)=O)CCNC1=O c1(C(=O)NCCC(C)N(C(=O)COCC2CCOC2)C)cccc2cc[nH]c12 c12cc(F)ccc1NC2.C1(C(F)F)(CC)CC(c2nnnn2CCCF)(OC)C1 c1(C(N2CC(N(C)C(c3nsnc3O)=O)C2)=O)cccn(C2CC2)c1=O CC1(C)CCN(C(C2(C)CCNC2=O)=O)CC1C(=O)NCC1CC(C#N)C1 CCCCC(CC)CCC(=O)N(CCNC(C1CCCCC1F)=O)C1CC1 c1(C(=O)NCCC2CC(Nc3nc(O)n(C)c(=O)c3)C2)noc2c1CCCCC2 C1(=O)CCCN1.C1(C(C)C(=O)NC2CN(C(=O)CN(C)C)C2)CCC(=O)N1 c1(CN(C(=O)CC2CCN2C(=O)C(O)Cc2ccccc2)CC)nncn1C C=C=CC(C)C(=O)NC1(c2ccccc2)CC(NC(=O)C(O)CC2CCCC2)C1 NS(=O)(=O)CCCC(=O)N1CCCC1C1(NC(C23CSC(C2)C3)=O)CC1 N1(C(c2ccc(OCC)cc2)=O)CCC(C)C(NC(c2ccnc(O)c2)=O)C1C c1(C(C(C)C)NC(CC2CC(OC(C)C)C2(C)C)=O)nnc2ccccn12 C#CCC(C)(C)C(=O)NCC(N1CCN(C(C2CCCSC2C)=O)CC1)C c1(CSC)cccc(C(N2CCC(C)(NC(=O)CC3CCC(C(N)=O)O3)C2)=O)c1 Cc1cc(C(=O)NC2C3CN(C(c4cnn5cccnc45)=O)CC23)c(I)cc1F C1CCCN(C)C(=O)N1.C(C(F)=C(C)C)SC.C1CN1 Nc1cc(Cl)ccc1C(N1CCN(C(c2csc(-c3ccoc3)n2)=O)C2CC12)=O c1(NC(c2cccc(C)c2C(F)(F)F)=O)cc(CO)c2c(c1)OC(F)(F)O2 c1(OC)ccc2[nH]c(=NC(C)C3CN(C(C4(C)C=CCCC4)=O)CCO3)sc2n1 c1(SC)ccc(C=CC(=O)N(C(C)CCNC(C2C(C)C2(F)F)=O)C)cc1 Cc1ccc(O)cc1C(=O)NCCCCCCNC(c1cnns1)=O Cc1nn(C)cc1C(N1CCC1CNC(c1csc(N2CCOCC2)n1)=O)=O C(Cc1nc(-c2cccs2)no1)(C(O)C(F)(F)F)C(c1ccc(F)cn1)C.N N1(C(c2n(C=C)ncc2)=O)CCN(C(=O)CC2CCC(=O)NC2)C(C(F)F)C1 N1(C(c2cc(C)n(C)c2)=O)CCC2CCN(C(C3(C)CCCCCC3)=O)CC2C1 C(=O)(C(CCNC(C1(CCOC)CC1)=O)OC)NCC=C CC(N=c1[nH]c2c(c(=NC3CCC(F)CC3)[nH]1)CCC2)c1ccc(Br)s1 C(=O)(C1CCCc2sccc21)NCCC1(OC)CN(C(=O)CC2CS(=O)(=O)C2)C1 C1(C(=O)OC)CCC(CNC(C2(C)OCCO2)c2nnnn2C2CCC2)O1 N1(C(C=Cc2c(C)nccc2)=O)CC2(CCCC2NC(c2nc(=N)cc[nH]2)=O)C1 c1(C(N(CCCCCNC(Cc2c(C)n(C)cn2)=O)C)=O)ccn2cccc2c1 c1(C(=O)NCC(CN(C(C2C(=C)C2)=O)C)(C)C)ccc(-n2ccnc2C)nc1 c1(OC)oc(C)nc1C(=O)N(CC(O)CNC(=O)CCc1ccccc1F)C N1(C(C)=O)CCC(C)(C(N2CCC(Cn3cc(CNS(N)(=O)=O)nn3)CC2)=O)C1 N1(C(C(C)=C2CCC2)=O)CC2(CCC2)CC1C(=O)NC(C(C)C)C1CCC1 N1(C(C(CC=C)(F)F)=O)CCC(CNC(c2ccc(Br)o2)=O)C(F)(F)C1 N1(C(C2(C)N(C(C3C(C)C3)=O)CC2)=O)CCC(F)(CO)CC1 CSC1=C(C(=O)N2CCN(C(=O)C(C3CCOCC3)O)C(CF)C2)CCCC1 c1(C(N(C2CCN(C(=O)C3=NNC(=O)C3)CC2)CC#C)=O)cc(Cl)c(C)cn1 c1(C(=O)NCCCC(C)C)cnn(CCNC(=O)CC2(CSC)CC2)c1 N1(C(C2(C)CCN(C(C(C)(C3CCC3)OC)=O)C2)=O)CC2CCCC(C2)C1 C(=O)(C(C(=O)N1CCC2(NC(c3c[nH]nc3CC)=O)CCCC12)C(C)C)OCC c1(C(N2CCC(C(C)NC(c3cn(CC)nn3)=O)CC2)=O)[nH]ccc(=O)c1C C12(NC(CC(c3ccccc3F)C)=O)CCCN(C(c3ccon3)=O)CC1C2 CN1CCc2[nH]c(=NCC3(C)CCN(C(c4cnc[nH]4)=O)C3)c(C#N)cc2C1 CCCCCC(O)C(=O)N1CCC(C(F)CNC(c2cccn2C2CC2)=O)CC1 c1(OC)ncnc(C)c1C(N1CCC2(CC2NC(=O)CC2CCCC2C)C1)=O N1(C(Cc2c(O)ccc(C)c2)=O)CCC2(CCN(Cc3cc(I)ccc3O)C2)C1 c1(NC(=O)CN2CCN(S(=O)(=O)C3CCCCC3)CC2)cc([N+](=O)[O-])ccn1 CCC1=C(C(=O)NC2(C(N3CCOC4(CCCC4)C3)=O)CC(F)C2)CCCO1 N1(C(C2(C#C)CCC2)=O)C2CCC1CC(F)(CNC(=O)C(C)(C)C(=C)Cl)C2 CN1CCC(CNC(=O)COc2ccccc2I)CC1=O C1(NC(Cc2c(C)ocn2)=O)CN(C(=O)C(C)C2CC2)C2(CCCC2)C1 N1(C(CCN(C(C)=O)C)=O)CCN(C2CCN(C(=O)C(C)n3cccc3)C2)CC1 CCCC(CCC)C(=O)N1CCN(C(c2cn(C3COC3)nn2)=O)C(COC)C1 N#Cc1cnc(NC2CCCN(CCNC(C3(CO)CC3)=O)C2)c(Br)c1 C(CCCCC(=O)N1CCCC(CN(C(=O)C(c2cccc(C)c2)C)C)C1)=CC CC1(C(=O)NCC2(CO)CCN(C(C3CC(C(F)(F)F)C3)=O)C2)CCC(=O)C1 C1(NC(C(C2CCCN(C(=O)C=Cc3ccoc3)C2)(C)C)=O)CC1C1CCCCC1 c1(C(=O)NC(C(=O)NCc2c(C)con2)CN(C)C)cc[nH]c(=N)n1 C1(C(=O)NC2C(NC(CCCOCC=C)=O)CCC2)CCNC(=O)C1 C(CC(=O)N=c1ccn(C(C)C)[nH]1)OCCCNC(C1(CC)CCCCCC1)=O C#CC1(F)CN(C(C2CCC2c2ccccc2Cl)=O)C1 CC(C)CC(O)C(C)C(=O)NCC1CC(C(=O)N(C)C(C)C)=NO1 C1(CC=C)(NC(c2csc(C)n2)=O)CCN(C(C2CC2C)=O)CC1 N1(C(C(N2CCC(C)CC2)=O)=O)CC(CNC(=O)CNc2nccs2)C2(CC2)C1 CC1COCC(CC(=O)NCC2CCC(C(=O)N(CCCC(F)(F)F)C)CC2)O1 C1(C(N2CCN(CCNC(C(OC)OC)=O)CC2)=O)CCC2CCC1O2 C12(CNC(C=CS(C)=O)=O)CCC(CC1)N2C(=O)CCC1CCCCC1 CCC(CO)(C(=O)NCC1CN(C(=O)C(c2cnn(C)c2)C)C(C)(C)C1)OC c1(N2C(CNC(CC(c3ccccc3)NC(N)=O)=O)CC2)ccc([N+](=O)[O-])cn1 C1(NC(C#CC(C)(C)C)=O)CCC2(CCN(C(C34CCCN3CCC4)=O)C2)C1 CN1CCN(C(C2CC(NC(c3cncc(Br)c3)=O)C2)=O)CC1CO CCC(CNC(=O)C=CC1CCCO1)(CC)NC(=O)Cc1cnn(C)n1 c1(OC)nccc(C(=O)NCC2CCC2C(N2CCOCC2CC(C)C)=O)n1 CC1CCN(C(=O)C(N2CCOCC2)=O)CCC1N1CC(c2ccccc2F)C1 C1(C(=O)NCC2C(CNC(c3c(-c4ccn(C)n4)n[nH]c3)=O)C2)CC2(CCC2)C1 c1(OC)nc(NC2CC(C)N(C(=O)CN3CCCCC3=O)C2)nc2[nH]cnc12 C(C)(C)(CCCC(=O)NC1(C(N)=O)CC1)NC(c1cc(C(C)=O)[nH]n1)=O CCCCCCOCC(=O)NCC(CNC(=O)C(C)COC)CO c1(OC)cc(C(=O)OC)ccc1NC(=O)CC1(N)CCOCC1 CC(CS(C)(=O)=O)C(=O)N1CC2CC1CC2NC(c1cc2ncccc2[nH]1)=O C1(C(=O)Nc2ccc(CNC(C(CC)SC)=O)cc2)CN2CCN1CC2C c1(C(N2CC(NC(CCCC#C)=O)CC3(C2)CC3)=O)c[nH]c2c(C#N)cccc12 CCCCC(C)(F)C(=O)NCC1CN(C(=O)CCCN2CCN(C(C)C)CC2)C1 c1(OC)ccc(C(N2CCC(c3ccccc3C)C2)C(=O)NC(C)C)cc1F C1(NC(C(C(COC)C)C)=O)CC2CC(C1)N(C(=O)C=C1CCC1)C2 C1(CNC(C2(C)CC(=C)C2)=O)CN(C(C2CC(n3ccnc3)C2)=O)CCC1C Cc1nc[nH]c1C(=O)NC1CCN(C(c2cc(CCCO)on2)=O)C1 c1(NC(C(=O)NC(c2ccn(C(C)C)n2)C)=O)cccc(-c2ccno2)c1 C12(C(=O)NC3CC4CN(C(c5nc(COC)oc5)=O)C3C4)CCC(CC1)C(C)O2 c1(C(=O)NCCCCC(C)NC(C2CC=C(C)CC2)=O)ccc2oncc2c1 C(=O)(C(C(C)(C)C)SC)NC1(CNC(CC(c2c(OC)cccc2)C)=O)CC1 N1(C(C2C(=C)CC2)=O)CCC(C2(NC(=O)C=CC3CCC3)CC2)C1 c1(CC(=O)NCC(C)NC(CSCC)=O)ccc(Cl)c(Br)c1 C(=O)(CCS(=O)(=O)CC(C)C)NC(CNC(CCC=CCC=C)=O)(C)C N1(C(CC2(CSC)CC2)=O)CC2CC(C(=O)NOCCC(F)(F)F)(C2)C1 C(=O)(C#CC1(C)CCCO1)N1CCCC(CNC(C(C(=C)Cl)(C)C)=O)(CO)C1 N1(C(C2(CN(C)C)CC2)=O)CCCC2(C1)C(NC(c1cn(C)nn1)=O)CCN2C C1(NC(Cn2c(C)cc(C)n2)=O)CCN(C(=O)CC(=O)Nc2nccs2)C(C)C1 c1(NC(CC(C)NC(Cc2cnc(C)s2)=O)C)nccc(C(F)(F)F)n1 c1(C(N2CCC(F)(CNC(C3(C=C)CCC3)=O)C2)=O)c[nH]cc(Cl)c1=O N12CCC(CC1C)C2.n1(CC)nccc1CN=CCC(=O)OC N1(C(C(C)c2ccco2)=O)CC(NC(=O)COCCC2CCCC2)CC1(C)C C1(CCC)(NC(=O)C(C)C(F)F)CCN(C(=O)Cc2ccc(F)c(C)c2)CC1 N1(C(C(CC=C)CNC(c2ccc[n+]([O-])c2)=O)=O)CC2(C)COCC2(C)C1 C(=O)(C1=CCCN(C(c2c(F)cc(Br)cc2F)=O)C1)Nc1ccc(OC)c(O)c1 N1(C(C(c2cn(C)nc2)NC(c2cccc(CO)n2)=O)=O)CCCC(C)(O)CC1 N1(C(C(C)N(CC)CC)=O)CC(C(=O)NC2(C(=O)N(C)C)CC2)C2(CC2)C1 C1(C(=O)NC(CC=C)CNC(C)=O)CN(C(=O)COC)c2ccccc2O1 c1(NC2C(=O)C2)ccccc1C(=O)NCC1(NC(=O)CCOCCCO)CC1 c1(OC)nccc(Cl)c1COC(c1nn(-c2cccc(C(F)(F)F)c2)cc1O)=O N1(CC)CCN(CCC(=O)N(CCNC(=O)COCc2scnc2C)CC)CC1 C1(CCNC(c2c(CC)non2)=O)CCCCN1C(C1CCC2(C1)N=N2)=O N1(C(CC(C)n2cccn2)=O)CCCCC1CCC(=O)Nc1c[nH]ccc1=O c1(OCCNC(=O)NC2CN(c3ccn(-c4ccccc4)n3)C2)ccc(F)cc1 CCCCCCCCC(F)C(=O)N1CC(NC(=O)Cn2ccccc2=O)C(F)C1 C1(NC(C2CCCCC2C(F)(F)F)=O)C2CC1N(C(C1CC=CCC1)=O)C2 c1(CC(=O)N(CCCOCCN(C(CCC#CC)=O)C)C)cccc(C)c1Cl C(=O)(CCC1=NNC(=O)CC1)N(C(C)CNC(=O)C(C1CCCCCC1)O)CC N1(C(c2c(F)cccc2F)=O)CCC2CCN(C(c3cscc3Cl)=O)CC2C1 C1(NC(c2cc(OC)cc(Br)c2)C)CCCC(C)(C)CC1 N1(Cc2c(C)cccn2)CC2CN(c3ncnc4n[nH]cc34)CC2C1 N12CCC3(CC1)CC3C(=O)N2CC(O)CO.c1(C(=O)O)c[nH]nc1-c1ccccc1 S(=O)(=O)(c1cc(CO)ccc1Br)N1C(C(N2CCc3ccnc(Cl)c3C2)=O)CC1 O=C(C1=CCSC1)NCC1(F)CC(NC(c2cscc2C(F)F)=O)C1 c1(C(N2CC(C)C(NC(c3cc(C#N)on3)=O)CC2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 Cc1cc2ncnc(N3CCSCC3CCNC(c3nn(C)cc3Cl)=O)c2[nH]1 N1(C(CCCc2n(C)cnn2)=O)CCC(NC(=O)COC2CCCC2)C12CC2 c1(NCCN(C(=O)OC)CC)[nH]c(=NCC2CCCC23CC3)nc2c1cnn2C c1(C(=O)NCCCC(C)NC(c2c(C)oc(C(C)C)c2)=O)nccc(Cl)c1O N1(C(c2cc(N)cc(O)n2)=O)CC2CC1CN(C(=O)CCSc1ccccc1)C2 Cc1ccc(C(N2CCCCC(NC(=O)C(O)c3ccco3)C2)=O)cc1N C(=O)(C#CC1CCCOC1)N1CC(CCNC(Cc2c(C)scc2)=O)OCC1 C1(NC(c2cn(CC)nc2C)=O)COC2(C1)CN(C(C1(Cl)CC1(F)F)=O)C2 Cc1nn(CC(=O)NC(C)CC(C)NC(C2(C(C)(F)F)CC2)=O)c(C)c1[N+](=O)[O-] c1(C(=O)NC(CN(C(C(CC=C)(F)F)=O)C)CC)c2c(cc3c1CCC3)CCC2 C(C)(CCCC(=O)N1CCc2n[nH]cc21)NC(CCN(CCC)C)=O c1(OC)c(C(N2CCN(CCN(C)C(C3(C)CC3(F)Cl)=O)CC2)=O)c(C)nn1C C12(NC(Cc3cc(C)[nH]n3)=O)CCCC1N(C(=O)C(c1cncc(F)c1)C)CC2 CC(C)(CCNC(C1CC1(F)Cl)=O)NC(=O)Cc1n[nH]cc1Br CCC(C)C(C(=O)NCCN1CCNC(=O)C1)NC(=O)C(C)CC#N C1(CC)CN(C(=O)CCOCCCNC(=O)C(C(C)OC)N(C)C)CCCO1 c1(CC(=O)N(CC(C)NC(=O)C(C)Cc2ccco2)CC)nc2c([nH]1)CCCC2 c1(C(=O)NCCCOC)ccc2c(n1)CN(C(c1cscc1C)=O)CC2 C(CC(C)C(=O)NCCC1(O)CN(C(c2sccc2CN(C)C)=O)C1)OC c1(C(N2CCC(C)C(N3CC(C)(CO)C3)CC2)=O)cn2cccc(Br)c2n1 c1(C(N(C(CNC(C2CCC(=O)N2)=O)C2CC2)C)=O)ccsc1Cl N1(C(c2nc(Br)cs2)=O)CC2C(C1)N2C(c1cnc(C(F)(F)F)nc1)=O C(CC(CO)C(C)C)NC(CN(C(c1ccc(SC)o1)=O)CC1CC1)=O C(=O)(N=c1cc(C2CC2)n(C)[nH]1)N1CCC(SC)C1C1Cc2ccccc2C1 C12(C(=O)NC(C)C(C)(C)O)CCC(CC1)N(C(=O)C(C)(C)N=[N+]=[N-])C2 CC1(NC(c2nncn2C2CC2)=O)CCCN(C(C2CC(O)C2)=O)C1 c1(OC)cc(C)ccc1OC1(NCC2CCCCC2)CCC1.C1CC1 CCC(CC)C(=O)NCCCC(C)(C)NC(C1C2CC(=O)CC12)=O C(CCC(C(=O)NCc1cnn(C)c1O)NC(=O)CC1CCCC12CC2)OC c1(C(N(C)CC2CCCN(C(C3CC(Cl)(Cl)C3)=O)C2)=O)nccc(Cl)c1O c1(OCC(=O)NCC(C)N(C(=O)Cc2cncc(C)c2)CC)c(Cl)cccc1Cl N1(C(c2cc(C)oc2)=O)CCCC(NC(c2ccc(Cl)c(C)c2)=O)C(F)C1 C(=O)(C(C)(O)CC)NCC(C1N(C(c2c(CC)nc[nH]2)=O)CCC1)(C)C c1(OCC)ccccc1C(=O)NC1CCC(NC(c2onc(CC)c2C)=O)C1 c1(C(N(CCCCNC(CCC#CC)=O)C)=O)cc(S(=O)(=O)C(C)C)ccc1F c1(C(N(C2CCN(C(=O)CSC(F)F)C2)CCC)=O)onc2c1CCCC2 c1(C(C(C)NC(=O)CCn2cc(C(c3ccccc3)O)nn2)C)ccc(Cl)cc1 N1(C(C(N)=O)C2CCCC2)CC23CCCC2(CN(C(c2ccc(Cl)cc2)=O)C3)C1 c1(C(N2CCCC(C)(NC(c3n(C)ccn3)=O)C2)=O)cc(F)c2[nH]nnc2c1 O=C1CCC(NC(=O)Nc2cccc(Cn3cccn3)c2)c2sccc2N1 c1(C(=O)OCC2CCC3CC3C2)cnc2c[nH]nc2c1 c1(C(N(CC(CC)NC(C2CCC2(C)C)=O)C)=O)cnc(O)cc1C c1(CN2CC3C(C(=O)Nc4cn[nH]c4)C3C2)cccc(F)c1Br Cc1cc(F)c(C(=O)NC2(C)CC(NC(=O)C(C3CCC(=O)N3)C)C2)cc1F N1(C(CNC(C(C)(C)C)=O)=O)CCC(=CCNC(C2C3CNC(=O)C23)=O)CC1 CC(C)C(C)C(CNC(=O)CS(C)(=O)=O)NC(=O)COCc1nccn1C C1(N(CC(O)Cc2ccccc2)CCOC)CCN(C(=O)C(C)CO)CC1 c1(C(N2C(COC(C)=O)CCCC2)C(=O)NC2CC2)ncc(Br)cc1F CC(C)CC(=O)NCC(=O)NC1CC1C(=O)NCC1OCC(OC(C)(C)C)C1 C1(C(=O)NCCc2nc(C)[nH]n2)CC(C)(C)CCN1C(=O)CC1C=CCCC1 CC1=CC(C(=O)NC(C)CCNC(C2CC2C(F)(F)F)=O)SC1 c1(CN2C(c3nc(C4CC4)no3)CC(OC)C2)ccc(O)cc1C N1(C(C(CSC)O)=O)CC(N(C(=O)CS(=O)(=O)N(C)C)C)C2(CC2)C1 C1(NC(c2c(C)cc[nH]2)=O)CCC2(C1)CN(C(c1cccc3ncnn13)=O)C2 Cc1oc(C(F)(F)F)c(C(=O)NCC2CCCN(C(c3c[nH]c(=N)o3)=O)C2)c1C C1(CC(=O)NCCCOCCN(C(C2C(=C)C2)=O)C)Cc2ccc(Cl)cc2C1=O c1(N2CCC(NC(C3(c4ccn(C)n4)CC3)=O)C2)ncc(S(C)(=O)=O)cc1Cl N1(C(c2c(OC)ccnc2)=O)CC(C)(C)CC1CC(=O)NOCC(O)C(C)C Cc1ccc(C(=O)NC(c2cnn(C)c2)C(=O)NCc2noc(C3CC3)n2)o1 C#CCC(O)C(=O)NC1(C(N2CCC(C)(CO)C2)=O)CCOCC1 CC(C)(C)C(C)(O)C(=O)NC1CC(F)(CNC(=O)CS(=O)(=O)C2CC2)C1 N1(C(c2c(C)nns2)=O)CC2CC2(C(=O)NC2CCCCC2)C1 C(C(=O)NCC1CC(O)CN1C(c1ccc(C(N)=O)[nH]1)=O)(C(C)(C)C)NC(C)=O C12(CNC(CC(=O)OC)=O)CC(NC(C3CCC(C(N)=O)O3)=O)(C1)C(C)O2 C=C=C(C)CC(=O)NCCCN(C(C1CC1c1sccc1C)=O)C(C)C C1(NC(C(CC)CCOC)=O)CN(C(c2ccc(N)c(F)c2)=O)C2(CCC2)C1 N1(C(c2c(CC)cno2)=O)CC(CNC(=O)Cc2cccnc2O)C(C)C1 c1(C(C2CC2)NC(=O)Nc2cccc(-c3ccno3)c2)nc2ccccc2s1 C(N=c1[nH]c(N2CC3CCC2C3)nc2ccsc12)c1snc(C)n1 c1(NCCC(CC)OC)cc(=NC(C)c2ccc[nH]2)[nH]c(C(C)C)n1 C#Cc1ccc(C(=O)NC2(CF)CCN(C(=O)C(c3nc(C)cs3)C)C2)nc1 C1(F)(C(=O)Nc2cccc(C3CC3)c2)CCCN(C(=O)C2CC2)C1 N12CCCCC(C1)C2=O.N1(CC(N2CC(N3CCNC3=O)C2)C)CSCC1=O CC1CC(CNC(=O)CCC2(C)N=N2)CCN1C(=O)CCC1CCCOC1 c1(NC23CC(C(=O)OC)(C2)C3)cc(=O)cc[nH]1.C12(C)CCN1ONC2=O c1(C(=O)NC(CC)CNC(=O)C(N)=O)cncc(Br)c1Cl c1(C(CNC(C(C)c2ncco2)=O)NC(=O)Cc2cncnc2)ccccc1F C12(C(N3CC(NC(c4nc(CCCC)sc4)=O)C(SC)C3)=O)CCCC1CCC2 N1(c2cc(NCC3CC(C(C)C)C3)ncn2)CC(C)OCC(C)(C)C1 C(=O)(C(C)CC(C)(C)C)NCC1(C(=O)NCC(C)CC2CCCC2)CC(=C)C1 CCCC(C(=O)NCC(C)NC(C1Cc2ccccc2C1)=O)S(N)(=O)=O C1(C)(CNC(Cc2n(C)ccn2)=O)CC(F)(F)CN1C(C1CCCC1O)=O C1(NC(CS(=O)(=O)N(C)C)=O)CCC2(CCN(C(c3ccccc3F)=O)CC2)C1 CC1(CNC(CC(C2CCC(CNC(C3CC3C(F)F)=O)CC2)=O)=O)CCOCC1 Cc1cc(C(N2CCC(NC(C34CC(C)(C3)OC4(C)C)=O)C2)=O)cc(C)c1Br Cc1ncccc1NC(C1CN(c2ncncc2F)C1)=O CC(C)(C)C(CNC(=O)C(O)c1ccsc1)C(=O)N1CC2(CC(F)C2)C1 C12(C(N(C)Cc3ccns3)=O)CC(CO)(CN1C(=O)CC1CCC3CC13)C2 C(CC(C)(c1nnnn1C1CCOCC1)NCC1CCCCO1)N(C)C C1(NC(=O)NCCN(CCOCC)C)CCCCC1 c1(NC(C2(c3cc[nH]n3)CC2)=O)ccc2cc(Br)cnc2n1 C(=O)(C1=CCC2(COC2)OC1)NC1C(CNC(CC2(C#N)CCCCC2)=O)CC1 C(CC(=O)N(C)Cc1nnc(C)o1)(C(C)CC)NC(C=CC(CC)C)=O c1(C(N2C(CNC(CNC(N)=O)=O)CC2)=O)ccc(N)c2ncccc12 c1(C(=O)NC2CC23CC(NC(C2(N4CCOC4=O)CC2)=O)C3)cc(F)cc(Cl)c1 C1(O)(CNC(C2(C)CC(C)C2)=O)CCN(C(=O)C(c2ccc(Cl)nc2)(F)F)CC1 C1(NC(C(CC=C)C)=O)C2CC1N(C(c1c(Cl)csc1Cl)=O)C2C C(=O)(C(C(C)C)C1CCC1)N1CCC(CN(C(C)C)C(c2n[nH]cc2Cl)=O)C1 C#CCC(C)(C(=O)NCC(C)N(C)C1CC1)NC(C1CCCC12CC2)=O C1(O)(CNC(CN(C)C2CC2)=O)CCCN(C(c2ncn(C)n2)=O)CC1 C1(CNC(CSCC#C)=O)C(C2CC2)CCN1C(=O)CCC(C)c1ccccc1 C=C(C)C1CN(C(C2CN(C(=O)C(C)CCN(C)C)CC23CCC3)=O)CCO1 c1(C(=O)OC)ncc[nH]c1=NC1CCN(C(=O)CC2(C)CCCO2)C1 c1(C(N(CC(O)CNC(c2ccsc2C#N)=O)C)=O)cc2cnccc2cc1F CC1CN(C(c2cccc(F)c2F)=O)CCN1C(=O)CN(C)C C1(CC(=O)N(C(CNC(=O)C=Cc2nccs2)C2CC2)C)CCCOC1 N1(C(C2(OC)CC2)=O)CC(C)(CCC(N2CCC(OC)C2)=O)C1 C#CCCCCC(=O)N1CC(CCNC(c2nc(C)n(C3CC3)c2C)=O)(OC)C1 N1(C(c2cc(C)c(C(=O)NC(C)(C)C)o2)=O)CC2CC(O)(C(F)(F)F)CC2C1 c1(C(=O)NCC2CCCCN(C(CC#N)=O)C2)nnn2c1CSCC2 N1(C(C(CC)OCC)=O)CCN(C(c2ccnc(C3CC3)c2)=O)CC1CC(F)F c1(NC(=O)OCC(N2CC(NC(CCC)=O)C2)=O)cn(C)nc1-c1ccncc1 N1(C(C=C(C)C(C)C)=O)CCCCC(C(=O)NCC2CCC(F)(F)C2)C1 C1(C(=O)NC(C2CN(C(c3ccncc3Cl)=O)C2)C)CCCC1(C)C c1(C(=O)NCCCOCCNC(c2c(C)ocn2)=O)cncc(Cl)c1 C1(C#N)(C(N2CCC(CN(C(C(C)C3CC3)=O)C)CC2)=O)CC2CC2C1 N#CC1(C(=O)NC2COCCC2NC(=O)COC2CCCCCC2)CC12CCC2 C(c1ccc(CNC2CC2C(=O)Nc2cccc(F)c2C(N)=O)cc1)=CC(=O)O C1(CNC(C(=O)NCCOCC(=O)NC2CC2)=O)CC1C1CCCC1 N1(C(CC(C)SC)=O)Cc2[nH]nc(C(N3CCC4(CCCC4)C3)=O)c2C1 N1(C(CCC2CCCN(C(C3CCC(N(C)C)C3)=O)C2)=O)CCCOC(C)(C)C1 C1(CCC(=O)N(C(C(=O)N(CCOC)CC)C)C2CC2)CCC(=O)C1 c1(C(C)=O)cccc(OC(C)C(=O)NC(C)CNC(c2conc2C)=O)c1 C(C1CCCCC1)=CC(=O)NC(C1CCN(C(C2C(Cl)(Cl)C23CC3)=O)CC1)C C1(C)(C(=O)NCc2cccc(C(=O)NCc3cc(C)c(C)s3)n2)CC2CCC1C2 N1(c2cc(C)c([N+](=O)[O-])cc2)CC2(C)CN(C(=O)Cn3cccn3)CC2(C)C1 CS(=O)c1ccccc1C(=O)NC1CC(O)(CNC(C23CC4CC2C3C4O)=O)C1 c1(C(CC2OCCN(C(C(C(=O)OC)C)=O)C2)=O)c([N+](=O)[O-])ccc(Cl)c1C CC1CN(C(C2CC2c2cccnc2)=O)CCCN1C(c1cc(C(F)F)n[nH]1)=O N(C1c2ccccc2CC1NC(C1(C)CCCCO1)=O)C(CCC(C)SC)=O C1(NC(c2ccc(C(C)C)o2)=O)CCN(C(C2CCN(C)CC2)=O)CC12CCC2 c1(N2CCN(CC(C)(C)NC(C3CCC(C)O3)=O)CC2)cccc(F)c1C#N N1(C(C23C(C)OC(C)(C2)C3)=O)CC(NC(c2cnnc(O)c2)=O)C2(CCC2)C1 N1(C(CSCCCC)=O)CCCC1C(C)NC(c1cnc(C(C)(C)C)o1)=O C12(C(=O)NCc3n(CC)c(C)nc3)CCC(N)(CC1)CC2 C1(CNC(c2cc(SC)c(C)o2)=O)CN(C(=O)CCc2ccc(C)o2)CCN1C c1(CCOC)ccc(S(=O)(=O)NC2CC2(c2cccc(C)c2)C)s1 N1(C(CCc2n(C)cnn2)=O)CCCC(C(=O)NCC2(O)CCC2)C1 c1(C(N2CCN(C(=O)Cc3ccon3)C3C2C3)=O)ccc2c(c1)CCC2 CCCC(CC)NC(c1cn(CC2CCCO2)nn1)c1nnnn1C(C)(C)C C1(C(=O)NC2(CC#C)CC2)(CNC(=O)CC(O)C2CCCC2)CCCO1 c1(C(N(C)CC2N(C(c3c(OC)n[nH]c3)=O)CCC2)=O)c(F)cccc1F N1(C(C2ON=C(CC)C2)=O)CCN(C(=O)COCC(C)C)CC(C)(F)C1 c1(C(C)C)ncncc1C(=O)N(CC(C)NC(C1CN(C)C1)=O)C c1(C(N2C(CNC(c3ccc(F)cc3F)=O)CC2)=O)cc(Cl)cc2c1CCC2 c1(OC)cc(F)ccc1CN1C(C(=O)NCC(c2ccccc2)=O)CC(OC)C1 c1(-n2cc(SCC3N(C(C4C(SCC)CCC4)=O)CCC3)nn2)cc(C)cc(F)c1 C(C(=O)NCC=CBr)(C1CCOC1)NC(=O)CSCC(F)F c1(C(C)C)cc(C(N2CCC2C(=O)NCCCN2CCCC2)=O)n(C)n1 C(=O)(C1CCCc2sccc21)NC1CN(C(CCS(=O)(=O)NC)=O)CC2(C1)CC2 N1(C(c2nc(C#C)sc2)=O)CC(NC(=O)CC(=O)OC)CC12CCCCC2 N1(C(C2CC(C)(O)C2)=O)CCN(CCNC(=O)C(c2ccc(F)cc2)F)CC1 N1(CC(N2CCC(C#N)C2)=O)CCN(C(C2CC(=O)N(C(C)(C)C)C2)=O)CC1=O C#CCCC(=O)NCC1CCC(NC(c2ccnn2C(C)C)=O)C1 C(CNC(c1cnn[nH]1)=O)(CC(=O)NCC(CSC)OC)OC N1(C(c2cc(NC(C)=O)cc(Br)c2)=O)CCN(C(=O)COC(C)C)CCC1C N1(C(CC(CC)O)=O)CC2CCC1CN2c1nc(OC)ncc1F c1(OCC(N2CC(CNC(CCSCCC)=O)C2)=O)c(C)cccc1Cl C(C(C)CN=c1ccc(S(=O)(=O)N(C2CCN(C)C2)C)c[nH]1)OC N1(C(C(=O)Nc2c(C)scc2)=O)CC(N)CC(O)C1 Cc1nsc(Br)c1C(=O)NCC1CCN1C(c1cnco1)=O c1(C(=O)NC2C(NC(C(CC#C)C3CC3)=O)CCCC2)cccn2nncc12 c1(C(N(CC(CC)NC(C=C(CCC)C)=O)C)=O)cc(C)cc(O)n1 N1(C(CNC(N)=O)=O)CCC2(NC(=O)CCCc3nc(C(F)F)no3)CC2C1 c1(OCC(N2CCC(CN(C)C(C3CCC(=O)NC3)=O)C2)=O)cc(Cl)cc(Cl)c1 n1(-c2ccc(NC3CC(C)(C)CC(C)(C)C3)cc2)nc(O)c2ccccc12 C1(O)(CNC(C(C)=C2CCCC2)=O)CN(C(c2cnc(CC(C)(C)C)o2)=O)C1 C(CCN=c1[nH]c(N2CCCN(C(=O)CC)CC2)nc2cc[nH]c12)OCC N1(C(c2cc(C)nc(O)n2)=O)CCOC2(CCC(NC(=O)C#CC3CC3)CC2)C1 C1(C(=O)NCCS(CC)(=O)=O)CCCCN(C(C2CC(=O)NC(=O)C2)=O)C1 c1(C(=O)NCC(C)(C)CNC(C2(C)CCCOC2)=O)cc(C#N)ccc1O C1(NC(C2(CO)CCN(C(C(c3ccn(C)c3)C)=O)C2)=O)CC(F)(F)C1(C)C C(CNC(C1(C)CC(C)=NO1)=O)(CC(=O)NCC1CC=CC1)OC c1(OC)cc(C2CCCN2C(=O)C(=O)NC2CN(C(=O)OC(C)(C)C)C2)ccn1 C1(NC(=O)CONC(c2coc(C3CC3)c2)=O)CCCCCCC1 N1(C(C(C)Cc2ccco2)=O)CC(NC(=O)C2=CCC2)CC(C)(C)C1 c1(C(=O)NC2C(NC(C3(OC(C)C)CCC3)=O)CCC2)cc2cccc(Cl)c2o1 N1(C(COCCCC(C)C)=O)CCOCCC1C(=O)N(C)CCC1CN(C)C1 c1(C(=O)NCC(CC)NC(CC(=C)I)=O)ccn(C)c(=O)c1 C1(C#N)(C(=O)NCC(c2ccccc2)NC(CCCNC(C)=O)=O)CCCOC1 C1(NC(C2(COC)CCCC2)=O)CN(C(=O)COC(F)(F)F)Cc2ccnn2C1 Cc1nn2c(C(=O)NCC(C3CCCCC3)NC(=O)C(C)CF)c(C)nc2s1 N1(C(=O)Nc2cc(-n3cccc3)cc(Cl)c2)CCC(O)(C(=O)Oc2cccnc2)CC1 C(=O)(C(C)(F)C(=O)N1CC(CNC(=O)CN2CCOCC2)C(C)C1)OC N1(C(Cc2c(OC)cccc2)=O)CCC(CCNC(c2cnsc2C)=O)CC1C C1(NCC(=O)NCCNC(CC)=O)CCC1NC(=O)CCC1CCCC1 C1(OC)CC(NC(c2cc(C)c(F)cn2)=O)C12CCN(C(c1ccon1)=O)CC2 CCCCCCC(F)C(=O)NC1(CO)CCN(C(=O)C2=CCCCC2)C1 C(=O)(C(C)(O)CCN(C)C)NC(C)CCCCNC(=O)CCC1(C)CC1 c1(OCCCNC(CNC23CCC(N(C)C)(CC2)C3)=O)ccc([N+](=O)[O-])cc1 C=CCCCC(C1CC1)NC(=O)CC1CCCN(C(C2CCCC2O)=O)C1 c1(NC(N(C(c2ccc(F)cc2)CO)C)=O)cnc(Cl)cc1Cl Cc1ccnn1CC(N1CCCC1CNC(C1C2CCCC12)=O)=O C(=O)(C(C)C(C)C(C)(C)C)N1CC(CC(=O)NCC=CC(=O)NCCOC)C1 c1(C(N(CCC(=O)NCC(=O)OCC)C)=O)cc(NC)n[nH]1 c1(C(=O)NC2(C)CCCN(C(=O)CCc3cnoc3)C2)cnc2cccnc2c1 Cc1cccc(Br)c1C(=O)NCC1(C)CCN(C(c2c(C)ncn2O)=O)C1 c1(C(=O)NCCOCCN(C(CC(C(C)C)C)=O)C)cnn2c1OCCCC2 C1(C(=O)OCC)NC(=O)C2CCC1N2C(=O)Cc1ccnn1C1CCC1 c1(CC)noc(C)c1C(=O)NCC(C)(CO)NC(c1cc(C(C)C)no1)=O N1(C(C)=O)CC2CCCC2(Nc2cc(C#N)ncn2)C1 c1(C(=O)NCCC(C)NC(c2cn(CC)nn2)=O)coc2c1CCCC2 c1(C(C)C(=O)NC(CCOCOCC)C)ccncc1F.C(C)(C)(C)O C1(C(N2CCCC(NC(COC(C)=O)=O)C2)=O)CC(=O)c2cc(Cl)ccc2O1 C1(NC(c2ccc(COC)[nH]2)=O)CCOC(CNC(c2cc(C#N)on2)=O)C1 C1(NC(CC2(OC)CC2)=O)CN(C(C2CCCSC2)=O)CC1(C)C CONC(=O)C(=O)NCC1CCN1C(c1cc(C)c(SC)o1)=O N1(C(Cc2n(C)ccc2)=O)CCC(CCCNC(C2CCC23CCC3)=O)CC1 C(CC(C)(C)C)(C(=O)N1CCC(NC(=O)CCc2cc(C)[nH]n2)C1C(C)C)OC CC1CN(C(=O)CCc2ccsc2Cl)CCC1NC(=O)CCNC(=O)C(C)(C)C c1(CC)ccc(Cl)c(NC(C2CC(F)(F)CN2Cc2ccc(CO)cc2)=O)c1 CON1CCC(N(C)C(C2CC(NC(=O)CC3(C)CCOC3)C2(C)C)=O)CC1 C1(CNC(C2C(C)(C)C2(C)C)=O)C(C2CC2)CCN1C(C12CC(CO1)C2)=O C(CC(C)C(=O)NC(C1CCN(C(=O)CCc2nc(C)c(C)o2)CC1)CO)OC c1(C(=O)NCCCCCN(C)C(C2CSCCS2)=O)ccn2cncc2c1 C(=O)(C1=Cc2ccccc2C1O)NCC1(NC(C2(SC)CC2)=O)CCCCC1C c1(C(=O)NC2CN(C(C3CC(SC)C3)=O)CC2N=[N+]=[N-])cnc2[nH]nc(O)c2c1 C1(CNC(C2N(C(C)=O)CCCC2)=O)(NC(C2CC(F)C2)=O)CC2CCC1CC2 N1(CC(=O)NCC2(c3nn[nH]n3)CC2)CCC(c2ccccc2)(CO)CC1 C1(C)(NC(c2c(C)cn(C)c2)=O)CCN(C(=O)C(c2c(C)n[nH]c2C)C)CC1 N1(C(C2CC(C)(O)C2)=O)CCN(C(=O)CC2(C#N)CCOCC2)CC(O)C1 N1(C(c2ccc(C#N)s2)=O)CCOCC(C(=O)NOC2CC3CCC2C3)C1 C1(NC(=O)C(=Cc2ccccc2)F)CCN(C(C2CC23CCCC3)=O)CC1O C1(N(C(C(C)CC23CC(C2)C3)=O)C(=O)OC(C)(C)C)C2CCCCCC12 C1(NC(=O)CCCOc2cccnc2)C2CCN(C(C3(F)CCCCC3)=O)C12 C(C(C)(C(=O)N1CCC(CO)(CNC(C2C3CC4C(C3)C24)=O)C1)OC)OC N(C1CCCc2[nH]ccc21)Cc1cccc(C(N(C(C)C)C)=O)c1 N1(C(C2C(C)(C)CO2)=O)C2CCC(C2)C1CNC(c1n[nH]cc1C(F)(F)F)=O N1(C(C=CCCC)=O)CCC=C(C(=O)NCCCCCN(C)C)C1 CC(C)(CC(F)F)C(=O)N1CCCC(CNC(C2CCC(=O)C2)=O)C1 C(=O)(CC1=CCN(C(=O)C(C)C)CC1)NCc1c(C)nc(F)cc1 CCCC(O)C(=O)NCC1CC(NC(C2(CO)CC2)=O)C(O)C1 c1(CNC(C(C)c2ccsc2)=O)ncoc1C1CN(C(c2ccccc2)=O)C1 N1(C(C(CSC)(C)C)=O)CC(CNC(=O)CCc2ncccc2C)C2(CCC2)C1 N1(C(CC2CC(=O)C2)=O)CCCCCC1CNC(c1cccc(OCCF)n1)=O c1(CN(C(C(C)NS(CCCC)(=O)=O)=O)CC(=O)O)nnc2n1CCC2 N1(C(C2CC(OC)C2)=O)CCC(C)(CNC(C2(c3ccc(Br)cc3)CC2)=O)C1 C12CN(CC1CC1CCOC1C)C2=O.C(CC(=O)NCC1CCCO1)NC(CC)=O Cc1c(CC(=O)NC2CC(O)CN(C(=O)C(F)CC(C)C)C2)sc2ccccc12 C1(C(=O)NC2CC(CC)C2)CNC(=O)CN1C(=O)CNc1ncccn1 c1(C(N(CCN(CCCOC(CC)C)CC(=O)OC)CC)=O)ccc(F)cc1F N1(C(CCOCC(C)C)=O)CC(NC(=O)CSC2CCOC2=O)C(C(F)F)C1 C1(NC(C2(CC)CC2)=O)CC2CCC(C1)N2C(=O)C(C)OC N1(C(c2cc(C)sc2)=O)CC2(NC(=O)C(C)Cc3cccc(Cl)c3)CCC1C2 N1(C(CCC)=O)CCC(NC(=O)C(C(C)C)n2ccnc2)C2(CCC2)C1 c1(C(=O)NC2CC2CNC(C2CC2C(=O)NCCO)=O)ccnc(O)c1 N1(C(C#CCNC(C(c2ccccc2)C)=O)=O)CC2CC(O)CC2C1 c1(C(=O)NCC2N(C(CCC=C)=O)CCC2C)ccc(OC)nc1OC C1(CC)CCC(N=c2[nH]c3c(c(=NCCCNC(C)=O)[nH]2)CCC3)CC1 CC1(C)COCC(Cc2ccc(C(F)(F)F)nc2)N1Cc1ccc([N+](=O)[O-])cc1 c1(CC)ccc(Cl)cc1NC(C1CC2CC2N1C(c1cnc(O)nc1O)=O)=O C1(C(N2C(C)(C(=O)OC)CC2)=O)CC(C)(C)CN1C(c1cc(F)n(C)n1)=O Cc1cc(Br)cc(S(=O)(=O)NC2CN(C(C3(C)CCCCC3)=O)CC2C#N)c1 C1(C(N(CCCNC(C2(C#N)CCOCC2)=O)C)=O)CCc2ncccc2C1 C1(CCNC(c2c(C)[nH]cc2)=O)CN(C(=O)Cn2ncccc2=O)CCCO1 c1(NC(N2CCC(CCN(C)C)C2)=O)cc(CSc2ccc(Cl)cc2)ccc1O C12(NC(c3[nH]ccc3-c3ccccc3)=O)CC(C1)N(C(=O)CC1CCCO1)C2 N1(C(C(c2ccc(CC)cc2)(C)C)=O)CCCCC(CNC(c2cnsn2)=O)C1 c1(CCC(=O)NC(C2CN(C(=O)CSC(F)(F)F)CCO2)C)nnc(S)n1C C(=O)(C1=Cc2ccccc2C1C)NC1CN(C(CCN(CC(C(C)C)C)C)=O)C1 C(=O)(C(O)CC(C)(C)C)N1C(C)C(NC(=O)Cc2ccc(O)cn2)CC1 CCC(C)(C)CCNc1cc(NCC(c2ncc(C)s2)C)ncn1 N1(C(C#CC2(CC)COC2)=O)CCC2CCN(C(=O)Cc3ccsc3)CC12 c1(OC)ccc2[nH]cc(C(=O)NC3CC(C)CN(C(C4CC(C)(C)C4)=O)C3)c2c1 N1(C(C2(O)CCC(CC)C2)=O)CC2CC(C1)CN(C(=O)CCCC(N)=O)C2 c1(C(=O)NCCCN(C(C2C(C(=O)OC)C2)=O)CCO)occ2c1CCOC2 CCC(C)CC(=O)NCC1CCCN1C(=O)C=C(C)I C(CN=c1nc(N2CCC3C(CCCN3C(C)C)C2)c2c([nH]1)CCC2)=CC N1(C(Cc2cncc(C)c2)=O)CCC(NC(=O)C=CBr)C(O)C1 C(=O)(C1=COc2ccccc2O1)NCCCOC(=O)NC C1(C)(C(C)C)CCN(C(C2(CNC(=O)C(F)=CC3CC3)CC23CCC3)=O)CC1 N#CC1=C(C(=O)NC2CCCC2CC(N2CC(N3CCOCC3)C2)=O)CCC1 C1(C(N(C(C)CO)C2CC2)=O)CCCC1CNC(c1scnc1Cl)=O C1(NC(C=C(CC)CC)=O)CCC2CC1CN2C(c1ncn(C)n1)=O C1(C(=O)NCC2CCC3CN(C(=O)CNS(N)(=O)=O)CC23)CC2CCCCCC12 N1(C(CC)=O)CC2CCC1C(NC(=O)C(C)CSc1ccc(C)cc1)C2 CCCCC(C)(F)C(=O)NCC1(OC)CCN(C(c2cc3occc3s2)=O)CC1 c12ccc(cn1)C(=O)NC1CCN2C1.c1(NC(=O)N(CCO)C2CC2)ccccc1 C=CCC(C)(C)CNC(C1(NC(=O)CC2CCC(=O)NC2)CCSC1)=O C1(C(=O)NCCN(C)C)(NC(C=C(COC)C)=O)CCCC1C C1(N(C(=O)Cc2cc[nH]c2)CCC)CCN(C(=O)CCC2CC2)CC1 C#Cc1ccc(C(=O)NCC2CCN(C(=O)OC(C)(C)C)CC2C)c(Cl)c1 N(C1CS(=O)(=O)Cc2ccccc21)C(=O)NC(C)CC1CCOCC1 N(C1c2ccccc2CC1NC(=O)CC1CC2CC2C1)C(C(F)=CC)=O N1(C(C(C2CCN(C(c3cccs3)=O)C2)C)=O)CC2CCC(C1)C2O C1(C)(CN(C)C)CN(C(=O)CCC2(C)CN(C(C3CC(=O)CCO3)=O)C2)CCO1 C1(CC(=O)NCC2N(C(CNC(CCC)=O)=O)CC=C2)CCC(C(F)(F)F)CC1 c1(Cn2cc(C(C)(C)C)nn2)ccc(SC2CCCO2)cc1.C12(CC1)C(=O)N2 Cc1nc(C(=O)NC(C2CCCN(C(C3CC(N(C)C)C3)=O)C2)C)sc1C C1(NC(c2ccc3cnnn3c2)=O)CCN(C(C2C=CCCC2)=O)C12CCCC2 C(=O)(C#CCNC(=O)C(C)OC(C)C)N(C(C(C)SC)C)C N1(C(c2c(C)nc(C(C)C)s2)=O)CC2CCN(C(C3COC(=O)O3)=O)CC12 Cn1nc([N+](=O)[O-])cc1C(=O)NCC1CCCCC1NC(=O)CCC1OCCO1 C(CCCC(=O)N1CCC1Cn1cc(CC(C)(C)C)nn1)N(C(C)C)C Cc1ccc(C(C)Oc2ccccc2C(F)(F)F)cc1 C(C1=NOC2CN(C(=O)CCc3ccnn3C)CC12)NC(C(C(=C)C)(C)C)=O c1(C(N2CCC(NC(C3C(C)C3(F)F)=O)C(C)(C)C2)=O)cc2cccn2c(O)n1 Cc1nc(=N)[nH]c(=NC(C)C(C2CCCCC2)NC(c2cccn2C)=O)[nH]1 c1(NC(c2ccc(-c3c(OC)cnc(F)c3)cc2)=O)cc(O)nc(=O)n1C N1(C(CN(C(C)=O)C)=O)CC2CC1CC2NC(=O)CN1CCCS1(=O)=O C1(N(C(=O)CCC2(C#N)CCC2)CC)CCCN(C(=O)C(C)c2ccsn2)CC1 N1(C(C2(SC)CC(=O)C2)=O)CCCC(C(N2CCC2C2CCC2)=O)CC1 N1(C(C2C(C)(COC)C2)=O)CC2CCC1C1CN(C(=O)CCN3CCCC3)CC21 C12(CNC(c3cc(SC)oc3C)=O)CCCCC1N(C(=O)C1=COCCC1)CC2 c1(C(=O)NC(C)C=CC(=O)NC2CCNC2=O)ccc2c(c1)CC2 CC1CCc2c(C(=O)NCC(CNC(c3cncn3C(C)C)=O)CO)csc2C1 C1(C)(C(=O)NC(CCOC)CNC(c2cc(C)nn2C2CC2)=O)CCNC(=O)C1 C1(CNC(C(CC)SC)=O)CN(C(=O)CC2(O)CCCCC2)C2COCC2O1 c1(C(=O)NCCC2(OCC)CN(C(=O)C(CCOC)OC)C2)ccc(F)cc1 c1(C(N(CCCN(C(CC(=O)NCC#C)=O)C)C)=O)c[nH]c(=O)c2ccnn12 c1(-c2scc(C(=O)NC3C(NC(CCSCC)=O)CCC3)n2)ccc(F)c(F)c1 c1(C(N(CC(C)NC(=O)CC(C)(O)C2CC2)C)=O)cccn2nnnc12 c1(CC)nn(C)c(CC(=O)N(CCCN(C)C(c2sc(=N)[nH]c2CC)=O)C)c1Cl c1(NC(=O)NC(CC)C(F)(F)F)cc(-c2cnn(CCF)c2)nc2ccccc12 CC1(C)CC(NC(C2(C)CC2(F)Cl)=O)CN(C(c2cccnc2Cl)=O)C1 N1(C(c2c(C)oc(CNC(c3cc(N)cc(F)c3)=O)n2)=O)CC(C)CCC1C c1(C(=O)NC2(C)CC2)cccc(C2CC2)c1.C(=O)(CSN)N(C)CCN c1(C(=O)NCC(CC(C)C)NC(c2cnc3n2CCS3)=O)ccc(F)cc1C#N CC1(C)CCC(C(=O)NC2CCCC2NC(c2cc(N(C)C)nc(Cl)c2)=O)CC1 c1(CNC(N(C(c2ccccc2)C(N)=O)C)=O)cnn(Cc2ccsc2)c1 CCCCCCC(F)C(=O)NCCC1CCCN(C(=O)CNc2ccccc2)C1 C1(NC(c2cc(C)ncc2C)=O)CC2CCC1C(NC(C1COCCOC1)=O)C2 c1(C(N2CCCC23CC3)C(=O)NC2(C)CC2)ccc(Cc2nnn(C)n2)cc1 C1(C(=O)NC2(CC3CC3)CCOCC2)(CNC(C2CCS(=O)(=O)N2)=O)CC(F)(F)C1 CC1CN(C(c2cc(O)cc(=O)o2)=O)CCN(C(C2CC(C3CC3)C2)=O)C1 C1(CNC(C2C(C)(Br)C2)=O)CC2(CCN(C(C3(C#N)CCCC3)=O)C2)CO1 c1(NC(CNC(C(C)=C(CC)C)=O)C2CCC2)ncccc1C(=O)OC C(=O)(C(Cc1ccccc1)S(C)(=O)=O)NCCNC(C(c1cncc(F)c1)C)=O c1(OC)ccc(NC(=O)CCS(C)=O)c2ccccc12 Cc1ccc(CNc2cnc(Cl)cc2C(N2CCCC2C(N)=O)=O)c(Cl)c1 N1(C(C(C(C)(C)C)n2cc(CC(C)(C)N(C)C)nn2)=O)CC2(CCC(=O)NC2)C1 c1(CNC(Cc2snc(CC)n2)=O)nccc(Cl)c1F c1(N2CCC(CCNC(c3c(C)cccn3)=O)C2)nnccc1C#N C(C)(CCC(=O)N1CCC(NC(C23CC(C(C)(F)F)(C2)C3)=O)C1)OC NC1CC(NCc2cnn(C3CCCCC3)c2)C12CCOCC2 N1(C(c2sc(CC)c(C)c2)=O)CCN(C(C2CCCC(=O)O2)=O)CC2(CC2)C1 c1(OC)cnc(N(C2CCN(c3ccc(Cl)cc3)C2=O)C)nc1C C#CC1CCCC1NC(=O)C=CC1CCCN1C(=O)CCCN1CCCC1 C(=O)(CCCC(=O)N1CC2CC1CN2C(=O)C(C)(c1cccs1)N(C)C)N(C)C C1(CN(C(=O)Cc2nn(C)cc2Cl)CC)CCN(C(=O)C(C)SC)CC1 C1(CCN(C(CC)=O)CC(=O)NC(C)=O)CN(CC(=O)Oc2cccs2)CC1C CCC(C)C(COC)N=c1nc2c(cnn2C)c(NCC(C)(CO)OC)[nH]1 c1(NC2(CNC(=O)C=Cc3ncc[nH]3)CCC2)cc(C(N)=O)nc(Cl)n1 N1(C(C2C(OC)(OC)CC2)=O)CCC(C(=O)NC(C(=O)OC)C2CC2)C12CCC2 N1(C(CC2(CSC)CC2)=O)CC2CC2(NC(c2csc(C(F)F)n2)=O)C1 C(=O)(C(F)C(C)C(F)(F)F)N1C(CNC(c2c(CC)nn(C)c2)=O)CC(F)(F)C1 N1(C(C2(CCOC)CC2)=O)CCC(O)(CN(C(=O)C(C)C(C)O)C)CC1 Nc1cc(Cl)cc(Cl)c1C(N1CCCC(CNC(=O)Cn2nccn2)C1)=O c1(C(=O)NCC23COC(CF)(C2)C3)cnc2occc2c1.C12(CCC1)CC(=O)N2 N1(C(C2C(C(=O)OC)C2)=O)CCCC2(CCCN2C(=O)C(C)CSC)C1 N1(C(CC=C)=O)CCCC(C(=O)NC(C2CCN(C(=O)CN(CC)CC)CC2)C)C1 Cc1ccc(N(C(=O)C(F)C(C)CNC(=O)CCOCC(F)F)C)cc1F c1(C(N2CCOCC(NC(C3CC(=O)NC3)=O)C2)=O)nc2ccccn2c1F Cn1cc(Cl)c(C(=O)NC(C2COC(C)(C)C2)c2ccccc2)n1 N1(C(C2CN(C(C)=O)C2)=O)CCC2(C(=O)N)CC2C1.c1(-c2ccco2)cc[nH]n1 c1(-c2ccc(OC)c(CO)c2)c[nH]c2ccc(C(N3CCCCC3CO)=O)cc12 Cc1nc(O)c(C(=O)NCc2cn(-c3ccncc3)nn2)cc1-c1ccccc1 c1(CCNC2(c3n(CC=C)nnn3)CCC(C)(C)C2)noc2cc(F)ccc12 c1(C(N2CC(C)C(NC(C(F)=CC)=O)C(C)C2)=O)cc([N+](=O)[O-])c(N)cc1F c1(-c2cn(C(CC)CC)nn2)nnc2n1CCC2.C12CCC(CC1)OCCO2 CC(c1ccccc1Cl)=CC(=O)NCC1CCCN1C(c1n[nH]cc1C1CC1)=O C1(NC(C(C)N2CCC2)=O)CC2CC(NC(c3cnnc(O)c3)=O)CC2C1 N1(C(C2(C)CCC2)=O)CCCC(C2CCN(C(=O)C3Cc4ccccc43)CC2)C1 CC(CC(F)(F)F)N(C(=O)COCCNC(C1CCNC1=O)=O)C CC(CS(C)(=O)=O)C(=O)N1CC(CCO)(NC(c2cccc(F)c2O)=O)C1 c1(C(=O)NC2C(O)CCN(C(c3c(C(N)=O)coc3)=O)C2)ccc2cc[nH]c2c1 C1(C(N2C(CN(C(C(c3ccccc3Cl)C)=O)C)CCC2)=O)CCC(=O)N(C)C1 C1(C(=O)NC(CCC)C2CC2)(NC(C2CCC(C3CC3)C2)=O)CCC(C)(C)C1 CN1N=C(C(=O)NCC2CN(C(=O)CCF)C3COCC3O2)CCC1=O c1(C(N2CC(CNC(C(C)(C)NS(C)(=O)=O)=O)OCC2)=O)cc2c[nH]cnc-2n1 C1(CCOC)(NC(=O)CC(F)(F)F)CCN(C(=O)C(F)Cc2ccccc2)CC1 C(=O)(C(C)(C)CC(=O)NCC1(NC(c2nn(C)c(C)c2Cl)=O)CC1)OC N1(C(C(=O)Nc2ccc(CC)cc2)C)CCCC2(C1)CN(C)C(=O)O2 C1(NC(c2cn(C)nn2)=O)CCCC2CN(C(=O)CCCCN=[N+]=[N-])CC12 CC12CSCC1CN(C(C1(F)CCN(C(c3cccc(Cl)c3)=O)CC1)=O)C2 C#Cc1ccc(CC(N2CCC(CC(C)NC(C34CC(O)C3C4)=O)CC2)=O)cc1 C(=O)(CCS(N)(=O)=O)NC(C1(O)CCN(C(c2cncc(O)c2Cl)=O)CC1)C C(=O)(CC1CS(=O)(=O)c2ccccc21)N1C(CNC(=O)C2=C(Cl)CCC2)CC1 C12(CNC(C(C=CCCC)O)=O)CC(COC)(CN1C(=O)C(O)C(F)(F)F)C2 C1(NC(C(C)OCC)=O)CC(N=c2ccc([N+](=O)[O-])c(C(F)(F)F)[nH]2)C12CCC2 CCCCC(CC)CC(=O)NC(C)(C)C(C)NC(=O)CCc1cnc[nH]1 CCC(CC(=O)NCC(C1CC1)N(C)C(c1nc(Cl)cs1)=O)c1ccccc1 c1(OC(C)C)cccc(C(=O)NCCC(C)N(C)C(C2CC(C)(C(=O)O)C2)=O)c1 c1(C(=O)NCCNC(=O)CC2CCCCC23CC3)ccc2ccnn2c1 N1(C(Cn2cc(CNC(CC)=O)nn2)=O)CCc2cc(C3CC3)ccc21 C1(C)(C(N2CCCC(C)(NC(C3C4CCC3CC4)=O)C2)=O)CCCNS1(=O)=O N1(C(=O)OC)CSCC1C(N1CCC(NC(=O)Cc2ccccc2)C1)=O C(=O)(C(C)(F)C(=O)NCCC(O)CNC(=O)C(=O)NC(C)C)OCC c1(C(N(CC(C(=O)NC)C)C)=O)ncccc1NC(c1ccc(C)s1)=O c1(NC(C2C3CN(C(C4CC(C)(C)C4)=O)CC32)=O)cc(Br)c(O)c(Br)c1 c1(OCC(=O)OC)ccc(C(N2CC(Cc3cn[nH]c3)C(C)C2)=O)cc1OC c1(OCC(=O)N(C2CCN(C(=O)Cc3ccsc3Cl)CC2)C)cncc(Cl)n1 C1(C(=O)NCC2(CCNC(Cc3c(C)ccs3)=O)CC2)CCS(=O)(=O)C(C)C1 Cc1nc2n(n1)CCCC2NC(=NCC(C1CCCC1)C1CC1)NC1CC1 c1(C(N2CC3CCN(C(CCOCC#C)=O)C3C2)=O)cc2nc(Cl)ccc2o1 C1(CNC(Cc2cc(C)nn2C)=O)CCC12CN(C(c1c[nH]cc1C)=O)C2 N1(C(=O)Cc2cc[nH]n2)CCCC(C2CCN(c3nnc(C(F)F)s3)C2)C1 c1(OCC(=O)NC2CC(NC(=O)CCC3CCNC3=O)C2)ccc2c(c1)CCC2 C1(NC(C(N2C(CC(C)O)CCC2)=O)=O)CC2CCC1C2 c1(OC)ccc(C(=O)NC2CN(C(=O)CSC3CCCCO3)CC2C)cc1C C1(C#N)(C(=O)NC2CC(N(C(C(Br)=C(C)C)=O)C)C2)CCCO1 N1(C(CC(=O)OCCC(C)C)=O)CCC(C)(CNC(C2CC(=C3CCC3)C2)=O)C1 C1(CNC(C(C=CC)O)=O)CCCCN(C(c2nc(C)ncc2Cl)=O)C1 C1(NC(C=CC(C)(C)NC(C=CCOC)=O)=O)CC(C)(C)C1OC N1(C(C(C)SC)=O)CC(NC(=O)CN2CCCCS2(=O)=O)CC(F)C1 C1(C(=O)NCCC(=O)NCCC(F)(F)F)(OC)CCCOC1 Cc1cnc(NC(=O)NCC2CCC23CCCO3)nc1C c1(C(N2CCN(C(CCCC=C)=O)CC2CCC)=O)ncn2cc(Cl)ccc12 C=CC(CC)CC(=O)N1CC=CC1(C(=O)NC)COC c1(C(=O)NC2CN(C(CC3(CC)CC3)=O)CC2C)ccc2nnc(C(F)F)n2c1 C1(NC(C(c2ccc(Cl)cc2)C)=O)C=CCN(C(C2(F)CC=CC2)=O)C1 N1(C(c2cc(C(=O)OC)on2)=O)CC2(CCC2)CC1CNC(=O)C1=CCC(C)CC1 N1(C(C(C2CCCO2)NC(CCC#CC)=O)=O)CC2(CCC(C)OC2)C1 C1(NC(C2CCCOC2)=O)CCCCN(CCOc2ccc(Cl)cc2)C1 CC1(C(=O)NC2CC(NC(C3CCCN3C(=O)NC3CCCC3)=O)C2)CCCC1 Cn1[nH]c(C(=O)NC2CCC2CNC(c2cnn(-c3ccccc3)n2)=O)nc1=O C1(C(=O)NCCC(=O)NCC#C)CC(C)CN(C(c2sccc2CO)=O)C1 C=CCCCC(=O)N1CCCCC1CCCNC(=O)C(c1ccccc1)O C1(NC(CN(CCC)C)=O)C2CCN(C(c3ccc(O)c(CO)c3)=O)CCC12 C12(NC(C(c3ccccc3)NC(c3n(C=C)ncc3)=O)=O)CCCN(CCC1)C2 C1(CCC)(CO)CCN(C(=O)CC2CCN(CCCN(C)C)C2)CC1O C1(C(N2C(CN(C(c3cncs3)=O)CC)CCC2)=O)CCCCC12CCC2 Cc1nc(C(F)(F)F)c(C(=O)NCC2(CCNC(=O)Cc3cnsc3)CC2)n1O c1(CC)nc(C(=O)NCCCC2CC2CNC(=O)CC2(OC)CC2)c(Br)s1 CCC1=C(C(=O)NC2CCCCC2NC(C2(C)COC2)=O)CCCO1 C1(N(c2c(O)ccc(OC)c2)C(=O)CSC(=N)N)CCC12CCNCC2 C1(NC(C2C3CN(CC4CCCC=C4Br)CC23)=O)CCc2ccccc2C1 c1(-n2cc(C(=O)NC(CNC(c3ccoc3)=O)C3CC3)nn2)ccc(F)cc1 CC(CN=c1ncc([N+](=O)[O-])c[nH]1)NC(c1cccc(C(C)(C)C)n1)=O c1(C(=O)NCc2n(C)ccn2)ccc2c(c1)CCC2NC(C1(C)CC=CCO1)=O c1(CC)cccc2c(CC(N3CC(NC(=O)C(N)=O)C(C)(C)C3)=O)c[nH]c12 Oc1cc(-c2ccc(-c3ccc(N4CCNCC4)cc3)c(F)c2)cc(O)n1 C1(C(=O)NCCCn2ccnc2)CC(F)CCN1C(=O)CC1COCCO1 C(CCCOC)(C(=O)N1CCC(CC(F)F)C1)NC(c1c(C#C)c[nH]n1)=O C1(NC(c2scc(C(=O)OC)n2)c2nnnn2C2(C)CC2)CCC2(CCCC2)C1 C1(CN(C(=O)C(C)Cc2ccnn2C)CC)CCCN1C(=O)Cc1ccsn1 C1(C(=O)Nc2c(C(=O)NCC(N)=O)cc(Cl)cc2)CC(=O)N2CCCCC12 N1(c2c(Br)cnc(OC)n2)CCC(C2CC2)(CNC(=O)C=CC2CC2)C1 Cc1nc(N2CC=CC(NC(c3cc(O)no3)=O)C2)c(F)c(C)n1 C(CC(C(C)(C)C)NC(c1ccc(C#N)o1)=O)N(C)C(c1cnc(Cl)s1)=O Nc1c(C(=O)NC2CCC(NC(c3cscn3)=O)C2)cccc1Br c1(OC)ccccc1C=CC(=O)N(C)CC1CCN(C(c2cn(C)cc2C)=O)C1 N1(C(CCCNC(C)=O)=O)C(C)C2CC1C2NC(=O)C=C1CCC(C)CC1 c1(C(=O)OC)nsc(=NCCC2CCCN(C(=O)CSC(F)F)C2)[nH]1 C1(C)(C(=O)NC(CN(C(CN(C)CC)=O)C)C)CC1(Cl)Cl C1(CNC(CSCC=C)=O)CCN(C(=O)CN2CCCS2(=O)=O)CC1(F)F C(C(=O)NCCN(C(=O)COCC1(Cl)CC1)CC1CC1)N(CCOC)C C(=O)(CCCCC(C)(C)C)N(C)CC1(O)CCN(C(c2cc(Br)n[nH]2)=O)CC1 C1(CNC(C2C(CC)CCC2)=O)CC(F)(F)CN1C(=O)C(C)C(C)(F)F C12(C(=O)NC(C(C)C)(C)CNC(=O)CC(C)n3ccnc3)CCC(CC1)C2(C)C O=C(CCCC1CC1)NC1COCC1NC(=O)CCc1ccncc1 Cc1cc(C(=O)NC23CC2CN(C(=O)C(=O)C(C)(C)C)C3)cnc1C(F)F C1(NC(=O)CSc2n[nH]c(O)n2)CCN(C(C2CC(F)(F)C2)=O)CC1 N1(OC(c2cccc(-c3cnn(C)c3)c2)C2OCC(C)C2)CC2C(C(N)=O)C2C1 N1(C(c2occ(C)c2)=O)CC(C2CCCCN(C(C34CCC(C)(CO3)C4)=O)C2)C1 C12(NC(=O)Cc3cccnc3)CC3CCC(C1C2)N3C(c1cscc1C1CC1)=O c1(C(N2CCC(NC(C3C(COC)C3)=O)C2C)=O)cc2cc(Cl)ccc2o1 N1(C(CC(=O)NC2CC2)=O)CCN(C(C2CC3(CCCO3)C2)=O)CC2(CC2)C1 C(C(=O)N(C1CN(C(c2ccncc2-n2cccn2)=O)CC1O)C)(C(C)C)SC c1(OC)ccc(C)cc1-n1nnnc1SC.N12CC(C(O)C1)CS(N)(=O)=NC2=O c1(OC)cc(OC)cc(CCC(N2CCC(C)(NC(=O)CN3CC=CC3)C2)=O)c1 N1(C(C(C2CC2)OC)=O)CC(NC(c2cc(C(C)(F)F)ccc2C)=O)C2(CC2)C1 c1(CN(C2CCNCC23CC3)CC(N2CCCC2)=O)ccnc2ccccc12 CCC(CC)(C(=O)ON1CC(F)(F)C1C1CC1)OC.C1C(=O)NO1 N1(C(C2CC(CC)(CC)C2)=O)CCC(C)(C)C(CNC(=O)CC2CC(C)(C)C2)C1 c1(C(N2CCCC(CNC(c3c(CC)c[nH]c3)=O)CC2)=O)cccc2oncc12 C(CC(=O)Nc1cc(CO)cc(F)c1)(C(F)(F)F)NC(Cn1cnc(C#N)n1)=O N1(C(c2c(CC)c[nH]n2)=O)CC2CCC(C1)N(C(=O)Cc1ncoc1C)C2 C(=O)(CCCCC(C)=O)NC1C2OCC(C(=O)NCC(C(=O)NC)C)(C2)C1 c1(C(=O)NCC(C)N(C(=O)COc2cccc(C)c2)CC)ccc2ccnn2c1 N1(C(c2nc(C)c(C)s2)=O)CC(NCC(O)CN(C)C)OCC12CNC(=O)OC2 N1(C(CCSC)=O)CCN(C(=O)CCc2cc(C)no2)CC1CC(C)(C)C C(CC(C(=O)NC(c1ccccc1C)C)NC(c1cncc(O)c1)=O)=CC N1(C(C(=O)OCC)C)CCOCC(C(=O)NCCCN(C)C2CC2)C1 N1(C(C)=O)CC(NC(C2CCN(C(C3CN(C)C3)=O)CC2)=O)C(n2ccnn2)C1 C1(CCC(N2CCC(OCC)C2)=O)CCCN(C(c2cnc(C)s2)=O)C1 c1(SC)nc(C(=O)N(C(C(=O)O)C(C)O)C)cc(O)n1 c1(CNC(C(C)C(C)(C)C)c2nnnn2C2CCC2)cc2cc(Br)cc(F)c2o1 N12CCC(C1)NC(=O)CC2.C1(OCC)CC(C(=O)NCCOC(C)C)C1 Cc1n[nH]c(C)c1S(=O)(=O)N1CC(C(=O)N=c2cc(C)o[nH]2)C(C2CC2)C1 CC1=C(C(=O)N2CCCN(C(=O)C(c3ccccc3)F)CC2)COCC1 c1(OC)ccc(N)c(C(=O)NC2CCCC(N(C(=O)CNc3nccs3)C)C2)c1 c1(C(=O)NC(CNC(CC=C(C)C)=O)CO)cccc(Cn2cccn2)c1 c1(C(=O)NCC(C)N(C(c2cccc(N)n2)=O)CC)cc2sccc2s1 N1(C(Cc2n(C)c(C(F)(F)F)nn2)=O)CC2CC(C1)N(C(C1CCCO1)=O)C2 N1(C(c2c(COC)nn(C)c2)=O)C(C)CN(C(=O)C2=CCCC2)CC1C C=CCC(C)(C(=O)NC1CCN(C(=O)CSCC)CC1CC)N(C)C c1(C(N2C3CN(C(c4c(C)nsc4)=O)C(C3)C2)=O)cc(F)c(Br)c(F)c1 C1(NC(c2cccc(SCC#C)c2)=O)CCSC12CN(C(=O)C(O)C1CC1)C2 C(=O)(C(C)(C)c1nccs1)NCC1CN(C(C(C2CCCC2)NC(=O)OC)=O)C1 c1(CNC(c2cnsc2)=O)csc(CNC(=O)C(c2cccnc2)O)n1 C(=O)(C1=C(Cl)CCC(C)C1)NC(c1cccc(C)c1)CNC(C1(F)CC=CC1)=O c1(N2CCC(CC(=O)NCCC3CCCC3O)C2)cc(-c2ccccc2)ncn1 N1(C(C2CCC(OC)C2)=O)CC2CC(C(=O)NC(c3cncc(F)c3)C)(C2)C1 C1(C(N(C(C)CCNC(=O)Cc2ccccc2)C)=O)CCOCC12CCCCC2 C1(C(=O)NC2C(Nc3c(C#N)cncn3)CCCC2)CC2(C1)NC(=O)NC2=O CC1(CCNCCc2nc(C3CC3)no2)CC(=O)C1 N1(C(c2c(CC)csc2)=O)CCC(C(=O)NCC2(C)CC2(C)C)CC1(C)C c1(CCN2C(C(F)(F)F)CC(C(=O)OC)C2)ccc(C)cc1Cl C=C(C)CC(C(=O)NC1CCC(NC(C2C(C)C2C)=O)CC1)NC(C)=O C1(NC(C)=O)CCCC(NC(c2csc(Cc3ccc(F)cc3)n2)=O)C1 N1(C(C(CC(C)C)N(C(C2=CC(C)(CC)C2)=O)C)=O)CC(C2CCCC2)C1 C1(CN(C(C2C(=C)CC2)=O)C)C2CN(C(=O)Cc3cccc(COC)c3)CC12 CCCCCCCC(O)C(F)(F)C(=O)NC(C)CN(C)C(c1nnccc1C)=O Cc1nc(C(CO)NC(C2(C)CN(C(c3csnc3Cl)=O)C2)=O)n[nH]1 C(=O)(CCC(=O)NCC(c1cccc(Cl)c1)NC(C1CC(C)(F)C1)=O)OC C1(F)(CNC(C=Cc2n(C)ncc2)=O)CCN(C(C2CC2C(F)(F)F)=O)CC1 C1(C(N2CCC(OC)(CNC(c3cnn(C)c3F)=O)C2)=O)CC2C=CC1C21CC1 C#CCC(C)(CC)C(=O)N1CC2CC1C2C(=O)NCCCCCCCC C1(NC(C(C)C)=O)CN(C(c2cccc(-c3ccccc3F)c2)=O)CCC1F Cc1c(C(N2CCC(c3cnco3)C2)=O)oc(=O)c2ccccc12 N1(C(c2cncc(NC)c2)=O)CCN(C(=O)Cn2cnnc2)CC12CC2 C=CCC(CC(F)(F)F)NC(=O)Cc1csc(=NCc2ccccc2)[nH]1 C=CCC(CC(=O)NCCN1CCC(CO)C1)NC(c1c[nH]nc1[N+](=O)[O-])=O N1(C(C2CCOCC2)=O)CCN(c2cc(F)ncn2)C(c2cn[nH]c2)C1 C1(CC=C)(C(=O)OCC)CCN(C(=O)CCOCCSC)CC1.C1(C)C(=O)O1 c1(C(=O)NCC(CNC(c2c(C#C)c[nH]n2)=O)C)ccc(S(N)(=O)=O)s1 c1(C(N(c2ccnc(C#N)c2)c2nc(C)c(Br)s2)=O)cc2cc(Cl)c(Cl)cc2[nH]1 Cc1cc(CCC(N2CC3CC(NC(=O)C(F)n4ccnc4)C2C3)=O)cc(C)c1 c1(NC(Cc2nc(NC(C3N(C)CCC3)=O)sc2)=O)cc(Br)cnc1O C1(NC(C=CC=CC)=O)CCN(C(c2nccn2C)=O)C(C2CC2)C1 C1(NC(Cc2nc(C)oc2)=O)CCCC(NC(=O)CCC2CCCN2C)C1 N1(C(C(CCSC)O)=O)CCCC2(CCCN(C(=O)CCc3cncnc3)C2)C1 N1(C(NOCCN(C)C)=O)CCC(=O)CC1C1CC1 C(=O)(C(C)(C)CC(C)C)NCCN1CCN(C(C2CN(CC)C(=O)C2)=O)CC1 c1(C(=O)NCC2C3CN(C(C4C(CC)OCC4)=O)CC32)cnc2ncccc2c1 c1(C(N2CCC(NC(Cc3ncc(C)o3)=O)C(O)C2)=O)ccc2c(c1)nnn2C c1(C(=O)NC2C(c3n(C)ccn3)CN(C(=O)C3=CCC3)C2)cc(F)c(F)cc1N c12cnc(nc1C(C)C)SCC13CC2(C1)C3.C(=O)(C(O)CC(F)F)OCC Nc1c(C(N2CCCC2CNC(=O)CCC2CCCOC2)=O)cccc1[N+](=O)[O-] c1(C(=O)NCC(CN(C)C(C2(c3cccc(Cl)n3)CC2)=O)O)ccc([N+](=O)[O-])n1C C(=O)(C(CCF)NC(C1CCCO1)=O)N1CC(C)(CC=C)C1 C1(NC(C2N(C(C)=O)CSC2)=O)CCCN(C(c2scc(C)c2C)=O)CC1 C(C(O)(C(F)(F)F)n1cncn1)Oc1ccccc1O.Cc1cccc(C)n1 c1(N(CCN(C(c2cnn(CCC)c2C)=O)C(C)C)C)cc(Cl)nc(SC)n1 N1(C(c2cnc(C)[nH]2)C(=O)NCCCCCC)CCc2c(Cl)cc(F)cc2C1C C1(NC(C2CC(=C)C2)=O)CC12CC(NC(c1n[nH]cc1Cl)=O)C2 C1(CN(c2nc(=NCCC3CC3)[nH]c3c2CCC3)C)CCCC12CCOCC2 c1(C(N2CC3C(N(C(C(C)NS(CC)(=O)=O)=O)C)C3C2)=O)cc(Cl)ncc1O CC(C(F)(F)F)(C1CC1)NC(=O)NC(c1ccccc1)C(F)F c1(C(=O)NCCC2CC(NC(C3(CCC)CCC3)=O)C2)cccnc1C C(C)(c1cccs1)=CC(N1CC(CCNC(c2nc(CCCC)sc2)=O)C1)=O C(=O)(C1Cc2ccc(C)cc21)NC1CCN(C(C2(CCOC)CC2)=O)CC1 Cc1ccc(C(F)C(N2CC(NC(=O)C(C)N(C)C)C(C)C2)=O)cc1 c1(C(N(C)CC2(NC(c3ccc(C(F)F)o3)=O)CC2)=O)nnn(C)c1N C1(CC=C)(CNC2CC3OCCCC23)CCCNCC1 c1(C(c2nnnn2C2COC2)NCC=CCOC)cc(OC)cc(Br)c1 c1(C(=O)NCCNC(C2C(C)COC2)=O)ccnc(Cl)c1O C1(CCNC(C(CN(CC)CC)F)=O)CN(C(=O)C(C)(C)C(N)=O)CCCO1 c1(C(N2C(C(=O)NCC(CC)(C)CO)CCC2)=O)c(C)[nH]c(C)c1C N1(Cc2cn(-c3cccc(OC)n3)nn2)CCc2sc(S(N)(=O)=O)cc2C1 c1(C(N2C(C)CC(CNC(=O)C3=CCCOC3)CC2)=O)cnn2cccc2c1 c1(C(=O)OC)nc(C2CN(C(=O)C(CN(C)C)N(C)C)C2)no1.C(C)(C)C CC(C)(CC(=O)NCC1C2CN(C(c3ccc(CO)cc3)=O)CC12)CC(F)(F)F c1(C(=O)NC(CCNC(C(CC)NC(N)=O)=O)C)cc(Br)cc2c1OCC2 C1(CNC(c2c(Cl)cccc2Cl)=O)CC2(CCC2)CN1C(=O)COC1CC=CC1 c1(OC)cc(C(=O)NC2(c3ccccc3)CC2)cnc1-c1ccccc1C(C)=O N1(C(c2ccc(C(=O)OC)s2)=O)CCN(C(C2CCCN(C)C2)=O)C(C(C)C)C1 C1(NC(Cc2ncc(C)s2)=O)CCCC(NC(=O)CN(c2ccncc2)C)CC1 C1(C(=O)C(C(=O)OC)c2ccccc2)CCCCCC1CO.C#CCN C1(CCN(C)C(C2CCC(=O)N2C)=O)CCN(C(c2cnco2)=O)CC1 CCCCCCC(C)C(=O)N(C1CCCC1)CCNC(c1snc(Cl)c1Cl)=O N1(C(C(C(C)(C)O)(F)F)=O)CCN(C(C2C3C4CCC(C4)C23)=O)C2(CCC2)C1 C1(C)(C(=O)NC2C(C(C)C)C2)CCC(NC(c2ccn(C(C)(C)C)c2)=O)C1 N1(C(c2cnc(OCC)s2)=O)CCN(C(C23CC2COC3(C)C)=O)C(C)C1 C#CC1(C)CCN(C(=O)CN(C(=O)C(C)C2CCC2)C(C)C)CC1 c1(C(=O)NC2CC(CNC(c3c(CC)nco3)=O)C2)cc(N)cc([N+](=O)[O-])c1 N1(C(C(F)=CCC)=O)CC(C(=O)OC)c2cc(Br)ccc21 N1(C(CN(C(C(CC=CCC)C)=O)CC(C)C)=O)CCCCC(CO)C1 C1(CNC(C(CC)(F)F)=O)CN(C(C2NC(=O)C3CC23)=O)CC12CC2 N1(C(c2sccc2Cl)=O)CCC(N(C(=O)CCc2ccccc2)CCO)CC1 N1(C(C2C(c3ccc(C)cc3)C2)=O)CC2(CC(NC(C3(CF)CCC3)=O)CO2)C1 C1(O)(CNC(C(C)SCCCC)=O)CCCN(C(c2cccc(C)c2N)=O)C1 C(c1cncc(O)c1)=CC(=O)NCCC1(O)CN(C(C2C(CCC)C2)=O)C1 CC(CN(C)C)CC(=O)NC1(C(=O)NCC2CC(C#N)C2)CC1C Cc1nn(C)c(F)c1C(=O)NCC1CCC(C)CN1C(c1c[nH]c(C(N)=O)c1)=O C(=O)(C(C)C(C)O)NC(C)CNC(C1(C)CC1C(F)(F)F)=O c1(C(=O)OC)ncc(NC(N2CCC(c3ncncc3F)CC2)=O)cn1 Cc1cc(C(=O)NCCCC(=O)NCC2(C(C)C)CC2)c[nH]c1=N C1(NC(C(N)=O)=O)C=CC(C(=O)NCCC2CCOC2)C1 c1(C(C(=O)NC2CN(C(C3(SC)CC3)=O)CC2C)O)ccc(F)c(Cl)c1F c1(C(N2CCC(O)(C(C(=O)OCC)(F)F)C2)=O)c(Br)ccc(C)c1F C1(N(CCNC(C)=O)C)CCCN(C(=O)C(=O)NCC2CC(C)CO2)C1 c1(NCc2cn(C(C)C(=O)NC3C(C)(C)C3(C)C)nn2)cc(Cl)c(Cl)c(Cl)c1 CC1CC(NC2CN(C(=O)N(C)C)CC2C)CN(C(=O)OC(C)(C)C)C1 Cc1cc(C(=O)NCC(CNC(C2CCn3ncnc3C2)=O)CO)c(Cl)cc1F Cc1c(Br)sc(C(N2CC(O)(C(C)NC(C3C4COCC34)=O)C2)=O)c1C C1(C(=O)NC(C(C)O)C(=O)NC(C)Cc2cnn(C)c2)CC2CCC1CC2 C12(C(=O)OC)CCC(C(=O)NCC3(NC(=O)CC4CC4)CCCC3)(C1)OC2 c1(NC(C2CN(Cc3sc(Br)nc3Br)CCC2(F)F)=O)c(Cl)c(F)nc(F)c1Cl N1(C(COCC)=O)CC2(CCC2)CC1CNC(C1C(C)(C)OC1(C)C)=O C(C(F)(F)C(=O)NC1CCCC(NC(=O)C(C)Cc2cccc(Cl)c2)C1)OC N1(C(C)C)CCOC(C(=O)NCC(C(C)C)NC(=O)Cc2ccns2)C1 c1(C(=O)NC(C)CCNC(=O)C(=O)NCC2CC2)cc(-c2ccccc2)[nH]n1 c1(C(=O)NCC2N(C(CCCC=C)=O)CCOC2)cccc(C)c1[N+](=O)[O-] c1(C(=O)OC)cc(NC(=O)CNC(=O)Cc2ccccc2N(C)C)c(C)cc1Br CC1CC(NC(C2CC2C(F)F)=O)CN(C(=O)CC2CC=CCC2)C1 C1(N(C(CC(C)CF)=O)C)CN(C(C2CC=CC2)=O)CC1(C)C c1(CC)ccc(C(N2CCC(C(=O)N(C3CCN(CC)C3)C)(CO)C2)=O)cc1 Cc1ccnnc1C(=O)NC1CC(CNC(=O)CCN2CCCCC2)C1 c1(C(=O)NC(C2(O)CN(C(c3sc(CC)c(C)c3)=O)C2)C)ccc2ccnn2c1 N1(C(c2c(C)nc(CO)s2)=O)CC2(CCN(C(C3CC(=C4CC4)C3)=O)C2)C1 C1(CC(N2C3CN(C(=O)C4CC4)CC2CC3)=O)COc2ccccc2O1 c1(C(=O)NCC(=O)NCC(=O)NC(C#C)CC2CCCO2)nc(C)sc1C N1(C(c2c(CNC(CC3CCCC(C)C3)=O)occ2)=O)CCC12CCC(C)CC2 c1(C(=O)NC2C(CNC(c3c(C)cno3)=O)C2)c(NC(N)=O)sc(C)c1C c1(C(=O)NC(C)CC(C)NC(=O)Cn2ccnn2)ccc(C(F)F)c(F)c1 N1(C(c2cnc(C)[nH]2)=O)CC(NC(C2COCCN2C)=O)CC2(CCOCC2)C1 CC1=C(C(=O)NC2CCC(N(C(=O)CN(C)C)C)C2)CCO1 c1(-c2sc(NCc3cncc(C)n3)c(C)n2)c[nH]c2ncccc12 S(=O)(=O)(c1cn(C)c(C)n1)NCCC(=O)NC1CC(F)(CNC(C(C)OC)=O)C1 c1(C(N2CCC(N(CCC)C(C3CC3F)=O)C2)=O)cc(Br)c(C)cc1F Cc1cc(C)c(C(=O)NCCC2CCC(NC(C3(O)CCOCC3)=O)C2)c(=O)o1 N1(C(C(C)=CC)=O)CCC(CCNC(=O)COC2CCOC2)C(F)(F)CC1 c1(CC)c[nH]c(C(N2CCCC2C(C)(C)CNC(c2ocnc2C)=O)=O)c1 N1(C(C(C(=O)OC)OC)=O)CCC2CC2(NC(=O)CCNC(C)=O)CC1 Cc1cccc(-n2cc(C(=O)N(C(C)CNC(C3CCC(C)(C)C3)=O)C)nn2)c1 C1(Cn2cc(CONC(c3c(C(=O)NC)nsc3I)=O)nn2)CC(C)(C)C(=O)O1 C1(C2CCC2)(CNC(C(C)O)=O)CCN(C(C2CCCS(=O)(=O)C2)=O)CC1 c1(C(=O)NCc2c(C)nc(-c3cccc(F)c3)s2)ccc(F)c(Br)c1 C1(C(=O)NC(CC)COCC2CC2)OCCC1CNC(c1cc(C)[nH]n1)=O CCCC(C(=O)N1CCC1CNC(=O)CNC(=O)CNC(C)=O)C(C)C C(C)(C(CC(=O)N1CC(C)(C#N)C1)NC(c1cocc1C)=O)OC C1(NC(c2cc(OC)ns2)=O)CCCC(CNC(=O)CCc2cc(OC)no2)C1 c1(OC)ccc(CC(=O)NCCC(C)NC(c2cnoc2-c2ccc(C)o2)=O)cc1 N1(C(c2c(C)cc(C)nc2)=O)CCC2C(CCN2C(=O)Cc2cn(C)nc2Cl)C1 C=CCCCC(C(=O)NC(c1nn[nH]n1)C1CC1)NC(=O)C(CC)C(=O)OCC C(C(F)(F)CC(O)CO)N(C)C(=O)NCc1cncc2c1CCC2 C=C1COCCN(C(=O)C2=CCN(C(=O)CC(O)CN(C)C)C2)C1 CCCC(C(=O)NC1CC(CNC(C2(C(=O)N(C)C)CC2)=O)C1)N(C)C C1(C(=O)NCC2(NC(CCC=C=C)=O)CCOC2)COc2cc(OC)ccc2C1 C1(N(C(COCC(=C)C)=O)C)CCN(C(c2nccn3nccc23)=O)CC12CC2 c1(OCC=C)cccnc1C(=O)NCCCOCCCNC(C1CNC(=O)C1)=O N1(C(C2ON=C(C(C)C)C2)=O)CCC(C2CCN(Cc3cnn(C)n3)C2)CC1 c1(-c2n(-c3cncc(C)c3)nc(C(F)F)n2)c[nH]c2c(F)ccc(F)c2c1=O c1(C(N(C2CCN(C(=O)COc3ccccc3)C2)CCC)=O)ncccc1Cl c1(C(C)NC(c2c(CNC(c3cc(C)oc3)=O)cco2)=O)ncccc1C C=C=CCCC(=O)NC(C)C(C)(C)NC(C1CCCN(C(=O)C(C)COC)C1)=O c1(C(=O)NC(CCC)C)c2c(nn1C)CCN(C(c1cc(C)cc(C#N)c1)=O)C2 c1(CC)cc(C(=O)NC(CCC2CC2)C(=O)NC2CC2c2cccnc2)ncn1 c1(C(=O)NCC(CC)NC(C2CC(C)C2(C)C)=O)cnc(OC)nc1 C1(CC)CN(C(C2(C)CN(C(=O)CS(C)(=O)=O)CC2C)=O)CC(=O)N1 N1(C(C2CC(CC)(CC)C2)=O)CC(N(C)C(C2CCCN2C2CC2)=O)C2(CC2)C1 c1(C(=O)NCC2CCCN(C(=O)C(C3CCOCC3)O)C2)cc2c([nH]1)CCOC2 c1(C(n2c3cnc(s3)c2=O)=O)c(F)cc(Cl)cc1F.C12CCN(C1)C2=O.C(C)(=O)OC C(CC(=O)N1CCC(CN(C(=O)CSc2n[nH]c(C)n2)C)C1)(C(F)(F)F)OC C12(C(=O)NCC=CCSC)CCC(CN(C(=O)CCCCN(C)C)C1)C2 c1(OC)ccc2c(c1)CC(C(C)C)CN2C(=O)NCC1(c2ccccc2F)CC1 N(C(=NCC(C)(C)C)NC(CCOC(F)F)C(C(O)C(C)C)(CC)CC)C(CC)C n1(CCCC)cc(CNC(=O)NCC2CCC(NC)CC2)c(C)n1 CCC(O)C(F)(F)C(=O)N1CCC(NC(c2nc(Cl)sc2Cl)=O)C1 C1(F)(CNC(CCC2CC(OC)C2)=O)CC(NC(=O)CCCn2cccn2)C1 O=C(CCS(=O)(=O)C(F)(F)F)NC1CC(O)CN(C(c2ccsn2)=O)C1 Cc1cc(CCC(=O)NC2CN(C(c3ncn(C)n3)=O)CCC2C)cc(C)c1 n1(CC(N2CCC(C)(NC(=O)COC3CCOCC3)C2)=O)ncc(C#N)c1N N1(C(c2c(C)oc(Cl)n2)=O)CC(C2CC2)(C(=O)NCC2(C)CCCCO2)C1 C(C)(C)(CC(=O)NCCCN(C)C(c1cc(C(=O)OC)co1)=O)OC C1(C(=O)NC(C2CCOC2)C#C)(NC(C2CC(F)C(=O)N2)=O)CCN(C)C1 c1(C(N2CCC(CNC(C3CC3(Cl)Cl)=O)C23CC3)=O)ccnc2ncccc12 CC1(C)CN(C(C2CC3CCC2CC3)=O)CCC1C(=O)NCCN1CCOCC1 Cc1nc2cc(C(=O)NC3CC(O)CN(C(c4cnns4)=O)C3)ccc2s1 C1(C(=O)NCC(c2cnn(C)c2)C)CC2CC1CC2NC(c1cc(Cl)cs1)=O C(c1ccc([N+](=O)[O-])s1)=CC(=O)NCC12N(C(COCC=C)=O)CCC1CC2 C1(CNC(c2c(N)sc(C)c2C)=O)CC2CC(C1)N(C(=O)C=CCO)C2 O=C(CC1OCCc2ccccc21)NCC1CN(C(=O)C(O)C2CC2)CCCO1 C1(CNC(CN(C(=O)C(O)C(C)C)CCC)=O)CCC(C)(C)CO1 Cc1ncc(S(=O)(=O)C(=O)NCC2(CO)CC2c2cc(F)ccc2Cl)o1 N1(C(C2(CC3CC3)CCOCC2)=O)CCCC(OCc2sccc2Cl)C1 CC(C)CCC(F)C(=O)N1CC(C(=O)NC2CC3(C2)CC(C)(C)C3)C(C)C1 N1(C(CC(CCCC)NC(c2cc(C)nn2CC)=O)=O)CCC2CN(C)CCC12 CC(C)C(C#N)C(=O)NCC1CCCCN(C(c2ccsc2)=O)C1 c1(OC)cc(OC)c(C(N2CCC(C(C)NC(c3snnc3C)=O)C2)=O)cc1N CC1CCc2c(C(N3CC(O)(CCNC(=O)CCn4ccnc4)C3)=O)csc2C1 N1(C(C2C(=C)C2)=O)CCCC2C1CCCCN2C(=O)CC=CC(C)(C)C c1(C(=O)NCC2(O)CN(C(C3CSCC(=O)N3)=O)C2)cnn2ncccc12 C(=O)(CCCC(C)CC)NCC1(CO)N(C(C(CC(=C)C)OC)=O)CC=C1 N1(C(c2cc(SC)ncc2)=O)CCCC(C2CCN(C(C3(C)COC3)=O)CC2)C1 c1(C(=O)NC(C2C(C(=O)Nc3c(CC)n(CC)nc3)C2)C)c(OC)cccc1C c1(-c2cc(C3CN(C(=O)NCC(COC)CSC)C3)[nH]n2)nnc2n1CCC2 C1(C(N2C(CN(C(CCC(=O)NCC)=O)C)CCC2)=O)CC2C(C1)C2(C)C c1(C(N2CC3(CN(C(COCCCCC)=O)C3)C2)=O)cccn2nncc12 N1(C(CCCSC)=O)CCC(NC(C2(F)CC2c2ccccc2)=O)CC1 c1(CC(=O)NC(CNC(C2CC(CC)C2)=O)C2CCC2)ncoc1C C1(OCCC)CCCN(C(C2(NC(=O)CCCN(C)C)CCSC2)=O)C1 C12(C(=O)NC3C(C(=O)OCC)CC3)CCC(NC(c3c[nH]cc3CC)=O)(CC1)C2 S(=O)(=O)(c1ccc(NC(c2nccn2C)C)c(C#N)c1)NC(CCC)(C)CO C(=O)(C1=COCCC1)NC1CC(C(C)Nc2cc(-n3ccnc3)ncn2)C1 N1(C(C(C)=CC)=O)CC(NC(C2COC(=O)N2C)=O)C2(CC2)C1 C1(C(N(CC(=O)NCC2=CCCCC2)C2CC2)=O)CCCC2(CC2)C1 C1(NC(c2cnc(C)[nH]2)=O)CN(C(=O)CC2CCC(C)(O)CC2)C2(CCCC2)C1 C(C1CCCCCC1)=CC(=O)NCC1CCCCCN1C(C1CCCO1)=O c1(C(C)NCc2ccoc2C(=O)O)c(F)cccc1Br N1(C(CP(C)(C)=O)=O)CCC2CCC(C1)N2C(c1cccnc1-n1cccn1)=O C1(C#N)(C(N2CCCC(CN(C(C(COC)C)=O)C)C2)=O)CC2(CC2)C1 Cc1c(C(N2CC3(C2)CN(C(C2CCN(C)C2)=O)C3)=O)cccc1C#N C1(C(=O)NCc2c(C(N3C(C)(C(=O)OC)C=CC3)=O)con2)CC(C)CC(C)C1 C(CC(=O)NCC1(CO)CC1C(F)(F)F)N(C)C(C1CCCC1)=O C1(CN(S(Oc2c(OC)cccc2Br)(=O)=O)C)CC2CC1CC2(F)F N1(C(C2(O)CCCN(C(C)=O)C2)=O)CC2CC1CN(C(=O)CCCN(C)C)C2 c1(OCCc2ncn(C)n2)cc(F)c(Cl)cc1[N+](=O)[O-] Cc1cncc(CC(=O)NCCCCCN(C)C(C2CCC(C)C2)=O)c1 C(C)(C)(C(C)CC(=O)NCCOC)NC(COCC)=O C1(NC(CSSC)=O)CCN(C(c2sc(CO)nc2C)=O)C(C)C1 CCC(C)(C#N)C(=O)NCC1CCCCC1NC(c1ncccc1SC)=O Cc1ccc(C)c(C(=O)NCC2C3CC2N(C(=O)C(c2ccccc2)F)C3)c1 Cc1cc(F)ncc1C(=O)NCC1(O)CCN(C(=O)C(C2CCC(=O)N2)C)CC1 C1(N(C(COCC#C)=O)CC)CCCN(C(c2ccc(CO)cc2F)=O)CC1 Cc1nc(CNC(=O)CCNC(=O)CO)oc1C(=O)N(C)CC1OCCC1(C)C N1(C(C(c2cn(C)nn2)NC(COCCCCC)=O)=O)CCCC(CCCC)C1 CC1(C)CCC(NC(C2CCS(=O)(=O)C2)=O)C(CNC(=O)C(C)(C)F)C1 CN1CCN(C(c2ccncc2F)=O)CC1CNC(c1nccc(C(F)F)n1)=O c1(C(N2CC(F)CC(NC(C3(CC(C)C)CC3)=O)C2)=O)ccc2c(c1)nnn2C C1(C(N2CCC(NC(COCC#C)=O)C2C)=O)Cc2nccnc2C1 C(=O)(N=S1(=O)CCCNCC1)c1nc2c(s1)CC(N)CC2 S(=O)(=O)(CCC1CCc2ccccc21)NC(=O)C(F)(Cl)c1ccccc1 c1(SCC(=O)NC(CCNC(C2(COC)CCOC2)=O)C)cc(C)cc(C)c1 C(=O)(C(C(C)C)N(C)C)NCC(CNC(C=C(CC)CC)=O)(C)O C1(C(CNc2cn(CCNC(C(c3ccn(C)n3)C)=O)nc2)O)CC2C=CC1C2 C1(OC)CC(CNC(C2CC2(Cl)Cl)=O)N(C(C2CCOCC2)=O)C1 C(N=c1nnc(C)c(C)[nH]1)c1ccc(CNC(c2c(C)coc2)=O)cc1 C1(C(N2CCOCC(CNC(C(C)=CC)=O)C2)=O)Cc2cc(F)ccc2O1 C1(NC(CCC#C)=O)CCN(C(C2CCC(CCCCC)O2)=O)CC1O C1(OC)CN(C(=O)Cn2nnc(=N)[nH]2)CC1NC(C1(C)CC(F)C1)=O C(C(=O)NC(C)C)(C(CCC(=O)OCC)OC)N1CCN(CCOCC)CC1 C(=O)(CC(C(F)F)N1CCOCC1)N(CC)CC1CCCN1C(=O)COC(F)F c1(-n2cc(C(CC(C)C)O)nn2)cc(Cl)ccc1C(N1CCN(CCO)CC1)=O N1(C(C(CSC)O)=O)CCC(C(C)NC(=O)Cc2cc(C(F)(F)F)n[nH]2)CC1 N1(C(C(N2CC(C)C2)C)=O)CCOCCC1C(=O)NC1CC1c1ccco1 C1(NC(=O)NCC(C=CC)O)CCN(C(=O)NCc2ccccc2)CC1 Cc1cc(C(=O)NC2CCCC2C(=O)Nc2cc(Cl)ccc2F)nc(Cl)c1 N1(C(C)=O)CCOC(COCCS(=O)(=O)Cc2cn(CCCC(=O)O)nn2)C1 C1(C(=O)NC(C(C)NC(CCC#C)=O)(C)C)CCC(C)(C)CC1 c1(CC)cccc(C(=O)N(C)CC2CCCN(C(=O)CC3CC3)C2)c1N c1(C(=O)NC2C3(CCN(C(CN(C)C)=O)CC3)C2)cc(S(=O)(=O)N2CCC2)c[nH]1 C1(C(NOCC(N2C(CC(C)C)CC2)=O)=O)CC1C1(C)COC1 N1(C(C(C(CC)C)O)=O)CCCC2(C1)CN(C(c1ccc(CO)o1)=O)C2 C1(CSC)CC(N=c2[nH]c3c(c(=NCC4COC(C)(C)CO4)[nH]2)CCC3)C1 c1(C(=O)NCCCCNC(C(C(C)O)NC(=O)C2CC2)=O)ccc(S(C)(=O)=O)s1 Cc1c(CC(=O)NC(C2CCCCC2)C(=O)NC2(CN(C)C)CC2)ncn1C c1(CCNC(=O)NC(c2cnnn2C)C)cccc2c1OCCO2 C1(CCNC)CN(CC2CC2)CCN1c1nc(SC)ns1 C12(C(=O)NCCN(C(C(C)C3CC3)=O)CC(C)O)CC(CCO1)C2 c1(C(N(C2CCN(C(=O)CC3CC3)C2)CC)=O)ccc2c(n1)NCCO2 Cc1nnc2n1CC(C(=O)NCCCC(C)NC(=O)CCN(C)CCO)C2 n1(CCC(=O)NC2(CNC(C(C=C)(C)O)=O)CCC2)cc[nH]c(=O)c1=O CC1CC(C(N2CCCCC2C2(NC(=O)CSC3CC3)CC2)=O)CC(C)O1 C1(N(C(=O)Cc2cccc(C(N)=O)c2)CCC)CCNCCC1C C1(C(=O)NCC(CC)CCO)CCN(C(=O)CC2CSCCO2)O1 N1(C(CC2C(=O)NC(=N)S2)=O)CCN(C(c2ncccc2O)=O)C2CCCCC12 N1(C(c2cccc(NCC)c2)=O)CC2(C1)SCCC2NC(=O)CC1CCC2CC12 C1(C)(C(=O)OC)CC2(CC(NC(=O)NC(C)CN3CCSCC3)C2)C1 N1(C(=O)NC2CCN(CC)C2)CCC(O)(c2cccc(C(F)(F)F)c2)CC1 N1(C(c2nc(SC)sc2)=O)CCCCC1C(C)NC(c1ccc(C(N)=O)o1)=O c1(NC(c2ccc(I)c(OC(F)(F)F)c2)=O)c(O)ccc(F)c1F CCC(C)(CNC(=O)C(F)C(C)(C)O)C(=O)NC1CC1CNC(C1CC1)=O N1(c2cc(NCC3(c4ccccc4)CC(F)C3)nc(C)n2)CCn2ncnc2C1 c1(C(N2CC(NC(=O)CCc3ccnc(Cl)c3)C3C2C3)=O)cnc2n1CCOC2 C1(CNC(c2cc(COC)[nH]n2)=O)CC(C)CCN1C(c1[nH]c(C)nc1C)=O CC1C2CCCCC2CN1C(=O)C(CCC1CC1)NC(c1cnsc1)=O c1(C(N2CCC(C)(c3cc[nH]n3)C2)C(=O)NCC(=C)C)cc(CC)cnc1OC C(=O)(CCC(=O)N1CCOCC1)NCC(=O)NC(C)(C)C C(C1=CCCOC1)NC(C=CCN(C(CNC(CCC)=O)=O)C)=O C1(N(C(C(C(C)O)C)=O)C)CCCN(C(c2cccc(C3CCCC3)c2)=O)CC1 C1(C(=O)NCC(C)(C)NC(C(COC)C)=O)CC2(CCC2OC)C1 N1(C(c2c(C)n(C3CCC3)nc2)=O)CC(NC(=O)Cc2cnsc2)CCC1C c1(C(=O)NC2CCC(CC(=O)NCCC#N)CC2)cccc2c(O)cccc12 c1(C(c2ccccc2)OCCCN(C)N(C)C)cc(O)c2ccoc2c1 c1(Cn2cc(CCN(C)C(=O)COc3ccc(F)cc3)nn2)c(Br)cccc1Br c1(-c2c(C)occ2)nc(C2CCCn3ccnc32)n(-c2ccc(N(C)C)cc2)n1 C#CCC(C)C(=O)NCC1(F)CC(CNC(C2CC2C(=O)OC)=O)C1 c1(CCCC(=O)NC(C)(C)CCNC(=O)C=CCN2CCCC2)c(F)cccc1F C1(NC(c2cnn(C)c2Cl)=O)CCC2(CC1)CN(C(=O)CC(C)(F)F)CCO2 N1(C(C(C2CC2)OC)=O)CCCC1CN(C(=O)C(=O)N(C)C)C1CC1 C1(Sc2cncc(C(=O)O)c2)CC2(CCC2)C(=O)O1.C12(CC3(CCC3)C1)C(=O)N2 Nc1ccc(C(=O)NCC(CNC(=O)COCC2CC2)C(F)(F)F)c(Br)c1 c1(C(C)CC(=O)NCCOC2CN(C(=O)C=C3CCOCC3)C2)cccc(F)c1 c1(CC(=O)NCC2C(NC(CCc3cc(C)on3)=O)C2)cccc2nonc12 Cc1cc(C=CC(=O)NC2CC23CC(NC(=O)C(F)=CC2CC2)C3)ccc1F n1(CC(=O)NCC2C(NC(COCCOC)=O)C2)ncn2cccc2c1=O C1(CN(c2ccncc2)C(C)=O)CN(C(=O)CCC2CC2)CC1c1cncn1C c1(CC)cncc(C(N2CC3C(NC(c4nc(C5CC5)cs4)=O)C3C2)=O)n1 C1(C(N2CCC(OCCNC(CCCCSC)=O)C2)=O)CCC(O)CN1C c1(C(N2CCOCC2C(N2CCOC(C3CCCC3)C2)=O)=O)cc2n(n1)CCC2 C(C(O)C(=O)N(CCCNC(c1ccc(-c2ccccc2)o1)=O)CC)=CCCC Cc1cc(C(=O)N(CCCCN(C(=O)CC2CCC2C)C)C)ncc1F C1(C(=O)NC(c2cn(CCOC)nn2)C)(CCF)CCN(C(=O)OC)C1 N1(C(C(=O)Nc2ccc(-c3nn[nH]n3)cc2)=O)CCCC1C1CCCO1 Cc1cncc(C=CC(=O)NC(CNC(=O)C=Cc2csc(C)n2)C(C)C)c1 C(C)(N=c1[nH]c(COC)nc2c(C)csc12)C1CN(C(C2(COC)CCCO2)=O)C1 c1(-c2n(CCCC)ncc2)cc(C#N)ccc1F.N12CCC(C1)C2=O C(CC(O)CC(=O)NCC1CC2(CC2)CN1C(=O)Cc1csc(S)n1)SC c1(C(N2CC(F)(CNC(C(C)OC)=O)C2)=O)ncc2ccccc2c1N CC(C(=O)NC1CCCC(NC(C2(CC3CC3)CC2)=O)C1)C(C)O N1(C2CC2)CCOC(C)(CC(=O)NCc2c(CNC(=O)OC(C)(C)C)con2)C1 c1(C(C(=O)N(CCNC(C(CSC)C)=O)C(C)C)(F)F)ccccc1C#N C(CCC(O)C(=O)NCC(C)(O)C1CCCC1)NC(c1cc(C)ns1)=O c1(C(N2CCC3C(NC(CC(C)C)=O)C32)=O)cc(C(F)(F)F)c(Cl)cn1 CC1CN(C(=O)Cc2ccc(O)cn2)CC1NC(=O)C(C)(C)c1ccsc1 c1(NC2CCCC3CN(C(c4cc(C)sn4)=O)CC32)nc(Cl)nc2c1cnn2C C(C(=O)NNC(=O)CC(O)c1ccccc1)c1ccc(C)c(Br)c1 C12(C(N3CC(CN(C)C)OCC3)=O)CC(CO1)N(C(C1(CO)CC(C)(C)C1)=O)C2 N1(C(c2ccc(CC)[nH]2)=O)CC2CC(C1)N(C(c1nc3cccnc3s1)=O)C2 S(=O)(=O)(c1cnccc1N1CCCC1)N1CCC(C(=O)OC(C)C)C1 Cc1cc(C(=O)NCC2C(C)CCN2C(=O)CC2(C#N)CC2)c(O)c(C)c1 c1(C(=O)NC2(CCCNC(C(C3CCOCC3)C)=O)CC2)ccc(CO)c(F)c1 C1(CC=C)(NC(=O)C(C)C2CCC2)CCN(C(C2CC(F)(CF)C2)=O)C1 CCCC(C)(O)CC(=O)NC1CC(CNC(c2cncn(C)c2=O)=O)CC1O Cc1ccc(C(N2CC(C)C(C)(CNC(C3CCCCC3O)=O)C2)=O)c(O)n1 Cc1nn(C)c(C)c1S(=O)(=O)N1CC2(CC2C(=O)NCCCN2CCOCC2)C1 Cc1ccc2ccc(C(=O)NC3CN(C(=O)CSc4nccs4)CC3F)nc2c1 c1(C(N(CC(CN(C(C2N(CCC)CCCC2)=O)C)O)C)=O)cc(C)ccc1N N1(C(C(C)(C2(C)CC2)OC)=O)CCC12CN(C(=O)C1=CCSC1)C2 c1(OC)c(C(N2CC(CC(C)NC(=O)CC3CCC(C)CO3)C2)=O)csc1C C(=O)(CC(C(F)F)NC(c1ccc(F)cc1C)=O)NC(C(=O)OCC)CC N1(C(c2cc(C(C)C)nc(O)c2)=O)CC2CCN(C(C3CCNC3=O)=O)CC2C1 C1(C(N2CCC(CC)(CO)C2)=O)CC(O)CCN1C(=O)Cc1cnoc1 n1(CC)c(C)cc(C(N2CCN(C(=O)CCc3cn[nH]c3)CC2C2CC2)=O)c1C c1(CC)nc(N2CCCC(COC)(NC(C3CNC(=O)N3C)=O)C2)cc(C#N)n1 C(C(CNC(=O)C1=COCCC1)C(F)(F)F)NC(c1c(C(=O)OC)coc1)=O N1(CC)CCCC1C(N1CCC(CN(C(=O)CCNS(=O)(=O)CC)C)C1)=O c1(C(N2C(CCCNC(C(CC=CC)C)=O)CCCC2)=O)cc(OC)cc[n+]1[O-] C1(CN(C(CCNC(C2C(C)C2)=O)=O)C)CCN(C(C2C3COCC23)=O)CC1 C(=O)(CCCCC(F)(F)F)N(CC(O)CNC(=O)Cc1csc2nccn12)C c1(C(N2CCCC(C(C)NC(CCC(=C)Cl)=O)C2)=O)ccc(N)c([N+](=O)[O-])c1 C#Cc1cnn(CC(=O)NCCOC(C2CC2C#C)=O)c1 c1(C(N2CCC(NC(C3(NC(C)=O)CCCC3)=O)C2)=O)cnc(O)c(C)c1 c1(C(N2CCC(NC(c3c(COC)cccc3)=O)C2C)=O)cc(OC)nc(C)c1 CC(C)CC(CC(=O)NC1CN(C(=O)C=C2CCCC2)CC1O)CC(N)=O C1(CNC(C2N(CC)C(=O)CC2)=O)CCN(C(c2csc(COC)c2)=O)C1(C)C C1(O)(CCNC(C(c2ccc(Cl)cc2)CC)=O)CCCN(C(=O)C=CCF)C1 C(C(CNC(c1cn(C2CC2)nn1)=O)CO)NC(c1ccn(C2CC2(F)F)n1)=O CC1=NOC(C(=O)NCC2CCCN2C(c2ccccc2C(N)=O)=O)C1C C1(C(=O)NC2CCN(C(c3ncccn3)C)CC2O)Cc2cccnc2C1 C1(NC(c2ncc(C)cc2C)=O)CCCN(C(=O)C=C2CCCCC2)CCC1 O(NC(=O)C(C)C1CCN(C(C2(C)CCN(C)C2)=O)CC1)CCC(C)C c1(C(=O)NCCC2CCCN(C(CC(C)C(F)F)=O)C2)c[nH]c(=O)c2ccnn12 C(=O)(N=c1nc(NC(c2ccccc2)=O)[nH]n1C)C12C(C)(CSC1)C2 Cc1sc(C(=O)NCC2CCN2C(c2cccnn2)=O)c(Br)c1C c1(C(=O)NCC(C2CCCC2)NC(c2cc(COC)on2)=O)cc(C)cnc1F C(=O)(C(C(C)(C)C)NC(=O)C(Cn1cncn1)NC(=O)C1=CCCCC1)NC N1(C(c2c(O)ccc(C)n2)=O)CCCN(C(c2cncc(C)c2Cl)=O)CC1C CC(C)C(C)(CNC(=O)Cc1cccnc1Cl)NC(c1csc(C(F)(F)F)n1)=O c1(C(N2CC(NC(C3(O)CCC3)=O)CC(F)C2)=O)ccn2c(O)nnc2c1 n1(C(C(=O)NC2(CN(C(c3c(C)nc(O)[nH]3)=O)C)CC2)C)nc([N+](=O)[O-])cc1C Cc1cc(C(=O)NC2CC(NC(=O)CCC3CCC(=O)C3)C2)nc(O)n1 N1(C(CCc2cncc(C)c2)=O)CCCCC(NC(=O)CC(C)C(C)C)CC1 C1(OC)CN(C(=O)CNC2CC2)C2COCC12 c1(C2CC(=O)NC2)nnc(N2CCOCC2Cc2ccc(Cl)cc2)n1CC1CC1 Cc1cccc(C(N2CCC(C(F)C(=O)N3CC(N4CC(F)C4)C3)C2)=O)c1 C1(S(N)(=O)=O)(C(=O)NC2C3CC(NC(Cc4c(C)noc4C)=O)CC32)CCC1 N1(C(c2cccc(C)c2I)=O)CC23CCCCC2(C1)CN(C(c1cc[nH]n1)=O)C3 c1(C(=O)NC(C2OCCN(C(CC(=O)NCC)=O)C2)C)cc(C)cc(C)n1 c1(NC(C2(C)CCN(Cc3ncccc3C(=O)O)C2)=O)cc(F)c(F)cc1F Cc1c(N)ccc(C(N2CCCCC(N(C)C(c3cc(O)nn3C)=O)C2)=O)c1F CCCC(CC(C)C)C(=O)NCC1(CNC(=O)CNC(=O)NC)CC(F)(F)C1 C1(COC)CCN(C(c2cncc(CNC(=O)Cc3csc(C)c3)c2)=O)CC1 c1(C(N(CCN(C(=O)C(C)NS(=O)(=O)CC)CC)CC)=O)cccn2nccc12 C#CCCCCCCCC(=O)N1CCN(C(=O)CCC(=O)CC)CC1 C(=O)(CS(=O)(=O)N1CC2C(C(=O)NCC(c3ccc(OC)cc3)O)C2C1)OCC N1(C(C(COC)O)=O)CCC(C)(NC(c2ccccc2Br)=O)C1 c1(C(=O)NC(CN(C(C(C=C)O)=O)CC)C)ccc(SC)cc1 C12(CCNC(c3c(C)con3)=O)CCC(CC1)N(C(c1ccc(=O)oc1)=O)C2 N1(C(CCCCCCSC)=O)CCC2(CCC(NC(=O)CCc3cscn3)C2)C1 c1(CN(NC(CCN(C(CCC)C)C2CC2)=O)CC)ccc(COC)o1 N1(C(C(c2cccnc2)NC(C(C)NC=O)=O)=O)CCOC(C(C)(C)C)C1 CC1(C)COCC(CC(=O)NCCC2CC(NC(C3(C)CC(F)C3)=O)C2)O1 c1(C(=O)NCCCCC2CCN(C(c3n(C)ccn3)=O)CC2)ccc(F)cc1Cl c1(OC)cc(CNc2ccc(N3CCSC(C)(C)C3)cc2)ccc1C#N N1(C(c2cnc(C(C)C)s2)=O)CCN(C(=O)CC2(O)CCC2)C(C)C1C c1(CC)nc(C)ncc1C(=O)NCC1CN(C(c2ncc(Cl)cc2Cl)=O)C2CC12 C1(CNC(=O)C2=CCCO2)CN(C(=O)C=CI)CCCO1 CC(O)C(F)(F)C(=O)N1CC(C(C)NC(c2ccc(F)s2)=O)C1 N1(C(CN(C)CC)=O)CC2CC(NC(=O)CCC3CCCCN3C)C(C2)C1 c1(OC)ccnc(C(=O)NCC(C)(C(C)C)NC(C2CC(O)CN2C)=O)c1 c1(C(=O)NC(C2CCN(C(Cc3c(C)nc[nH]3)=O)CC2)C)cc(Cl)nnc1Cl N1(C(CN(CC)CC)=O)CCCC2(CNC(c3ccc(OC)nc3C)=O)CCCC12 N1(C(C2CCC(C)CC2)=O)CCCCC(NC(=O)C=Cc2ccc(N(C)C)cn2)C1 c1(CN=c2ccnc(N(CCC3CCC(C)CC3)C)[nH]2)c[nH]c2cc(Cl)ccc12 n1(CCOC)nc(C(=O)NCC2C(C)CCN2C(=O)CCS(C)(=O)=O)ccc1=O Cc1cccc(CNc2cccc(C(=O)NCC3CCS(=O)(=O)C3)c2)c1Br c1(N2CCC(CC=C(C)C)C2)nc2c(c(=NCCc3cn[nH]c3)[nH]1)SCC2 N1(C(c2cc(C)[nH]n2)=O)CC2(NC(=O)CC(C)c3ccncc3)CCC1CC2 C1(OCCNC(=O)NCC(C2CCCCO2)(C)C)CCCOC1 N1(C(C(C)(F)F)=O)CC2CCN(c3ncc(I)cn3)C2C1 C1(S(=O)(=O)c2ccccc2)(C(=O)NCC2(CC(C)C)N=N2)CCCC1 CCC(C)(COC)C(=O)N1CCC(CN(C(=O)CC2CCC(OC)CC2)CC)C1 c1(C(C(=O)NC(C)CNC(c2c[nH]nc2C(F)(F)F)=O)(F)F)ccc(Cl)nc1 N1(C(C(C2CCCN(C(=O)OC(C)(C)C)C2)(C)C)=O)CCCC(C2COC2)C1 C1(CCNC(C2C(CCOC)C2)=O)CN(C(=O)C(N2CCCCC2)C)CCO1 c1(CC)cccc(C(=O)NC(CNC(c2ccc(C3CCCO3)[nH]2)=O)CC)c1N C1(C)(CNC(C(CCC)NC(C)=O)=O)CCCN(C(c2occc2C)=O)C1 CCC(CC)CC(F)C(=O)N1CC(C(O)C(=O)NCC(C(F)(F)F)OC)C1 C1(NC(c2ccc(C)c(F)c2)=O)CCN(C(c2ccccc2)=O)CCC1CO CCC(F)(F)C(=O)NCC1C2CC1N(C(=O)C(c1cccc(F)c1)(C)O)C2 C(=O)(CC(C)C(F)F)N1CCC(CC(C)NC(c2cn(CCO)nn2)=O)CC1 C1(NC(CC2CC(CC)C2)=O)CCN(CCNC(=O)C(F)C2CCCC2)CC1 N1(C(c2n(CC#C)ccc2)=O)CCC(C)(CC(=O)NC2CCC(F)(F)C2)C1 C1(SCC)CCC(C(=O)NC2(C(N3CCCC3CN=[N+]=[N-])=O)CC2(C)C)CC1 CCCC(C(O)C(=O)N1CCC12CN(C)C2)NC(=O)C(C)(C(C)C)OC N1(C(c2cn(CC)nc2)=O)CCC(N=c2nc[nH]s2)C(CC)C1 N1(C(COCCCOC)=O)CCC(CNC(c2cnnc(O)c2)=O)C12CCC2 C#Cc1cc(NC(=O)Nc2ccc(CS(N)(=O)=O)cc2)ccc1C C(=O)(C1CN(C)C(=O)c2ccccc21)NC1CC(CNC(CC(C=C)(C)C)=O)C1 c1(C(C)NC(=O)NC(CCN(CC)CC)CO)cccnc1OC C1(C(=O)NC(C2(NC(=O)CCC(=O)N3CCC(O)CC3)CC2)C)CCSC(C)C1 N1(C(=O)NCCN(CC#C)CC)CCOCC1C1CCC1 C=C(CNC(=O)COCc1ccccn1)CCNC(C1C2COCC12)=O c1(C(=O)NCC(C)N(C)C(c2ccc(F)c(C(F)F)n2)=O)cc2n(c1)CCCC2 Cc1cnc(C(N2CCC(C)(C)C2C(=O)NOCC2CC2)=O)c(F)c1 c1(CC(N2C(CC)CN(Cc3cccnc3C)CC2)=O)[nH]nc2c(Cl)cccc12 Cc1cc(C)c(CNC(=O)C(C)CN(C(=O)CSc2cn[nH]c2)C)s1 C(=O)(CC(C(F)F)C(C)(C)C)NC1(CC=C)CCCN(C(=O)C=CC)C1 C(C)(C)(C(C)CC(=O)NCc1cc(Cl)ccn1)NC(c1n(CC#C)cnn1)=O Cn1nc(C(N2CC3CCCCC3(CN)C2)=O)c2ncccc12 c1(C(N2CCC(OCCNC(C(C(C)C)N(C)C)=O)C2)=O)c(O)cccc1F N1(C(C2(CNC(C3C=C(C)CS3)=O)CC23CCC3)=O)CCS(=O)C(C)C1 CC(C)CC(CNC(C1CN(CC(C)C)C1)=O)NC(C1CCCC1)=O C1(N(C(=O)C(C)=C(C)CC)CC#C)CCN(C(C2CC(CCO)C2)=O)CC1 Cc1nc[nH]c(=NCC2(C)CCN(C(C3(C)CCOC(C)C3)=O)CC2)c1F c1(CC)[nH]nc(C(=O)NC2CCC2NC(=O)CCF)c1[N+](=O)[O-] c1(OC2CCN(C(C(Cc3cc(C)no3)NC(C)=O)=O)C2)ccc(Cl)cc1 C1(NC(c2cn(C)nn2)=O)CC(NC(=O)CC2CCC(=O)N2)C12CCC2 CC1(NC(C2(F)CN(C(=O)CN3CC4CC4C3)C2)=O)CCNC1=O Cc1cccc(C)c1C(O)C(=O)NC1COCC1NC(=O)COc1ccccc1 O=S1(=O)C2=CNC=CC2=NC2CCOCC2SCC2(CCC2)N1.C1(CO)CC1 C(=O)(C1=C(C)OCCS1)N1CCCC(N(C(C2(C)CCC2C(=O)OC)=O)CC)C1 c1(C(=O)O)ccc(CCN2CCC(c3cscn3)CC2)nc1Cl c1(C(=O)NCCC2CN(C(CCC(=C)Br)=O)C2)cc(C#N)ccc1F C(=O)(CC(C)(C)CC(F)F)N1CC(N(C(=O)COCC2CCCOC2)C)C(O)C1 C(CCCCCC(=O)Nc1cccc(F)c1)c1n(C)nc(-c2ccc(Cl)cn2)n1 C(C#Cc1c[nH]nn1)N.C(=O)(C1=CC2CCC1C2)C(=O)C(c1ccc(Br)cc1)F n1(CC(=O)NCCN(C(=O)CC2CCC(O)C2)C)nnc(C2CC2)n1 C(CCC(C)C(=O)N(CC(=O)NC(C(C)C)C1CCC1)C)OC(C)=O Cc1[nH]c2ccccc2c1C(N1CCCC1C(N1CCS(=O)CC1)=O)=O C1(CC(=O)NCCC(O)CNC(=O)CSc2cccc(F)c2)CCCCC1O c1(C2C(C(N3C(C4(NC(c5ccsc5)=O)CC4)CCC3)=O)C2)ccc(O)nc1 N1(C(C2C(C)(C)C2)=O)CCC(CNC(=O)CC2(O)CCC2)C12CCC2 N1(C(C(C)(N(C(=O)C(O)CC(N)=O)C)C2CC2)=O)CCC(C(N)=O)C(C)(C)C1 C1(CNC(Cn2cc(C(C)=O)nn2)=O)CC(O)CN1C(C1CCCCC1)=O c1(C(=O)NC2C(NC(c3c(CC)noc3)=O)C2)cnn(C2CC2)c1OC C1(C(N(C)CC2(O)CCN(C(CC3CC(SC)C3)=O)C2)=O)CN(CP(C)(C)=O)C1 C1(CC)CNC(=O)CN1C(=O)C(C1CC1)NC(c1cnc(O)c(F)c1)=O C1(NC(c2ccccn2)=O)CN(c2ccc3nnnn3n2)CC2(CC2)C1 Cc1cc(C(N2CCC(Cn3cc(CN(C)Cc4nccs4)nn3)C2)=O)co1 c1(C(=O)NCCC2CC(NC(c3cccc(NCC)c3)=O)C2)n[nH]c2c1COC2 C=CC1(NC(C2CC(OCC)C(OC)C2)=O)CCCCC1.CCCN1CC1.C1CC1 C1(NC(CC=C(C)C)=O)CCN(C(c2ccc(-c3cccs3)cc2F)=O)CC1O c1(N(C2CC3CNC2C3)C(c2ccc(C)s2)=O)cccc(C)c1F C1(C2=NOCC2)C(=O)NC2CCCN1C2.n1(C(C)C)cc(N(CCC#N)C)cn1 C1(N)C2CC3CN(C(c4ccc(OC(F)F)cn4)=O)C1C3C2.NC(=O)C(=O)NC CC(F)(F)C(C)(C)CC(=O)N1CCCC1(C)CNC(=O)Cn1nccn1 C1(CNC(C2OCCN(CC)C2)=O)CN(C(c2cncn2C(C)C)=O)CC1(C)C N=c1[nH]nc(CC(N2CCCC2C2(NC(c3csc(Cl)c3)=O)CC2)=O)s1 Cc1cnc(C(C(=O)NC2CCC2)N(C)CCc2ccccn2)s1 C1(C)(NC(CC2C(C)C2)=O)CCN(C(C2CC(OC3CC3)C2)=O)C1 C(=O)(C(F)(F)C(F)F)N1CC(O)(C(C)NC(c2cc(-c3ccc(Cl)s3)on2)=O)C1 c1(C(=O)NC2CC(NC(c3c(=N)[nH]cnc3)=O)C2)cn(CC#N)c2ccccc12 C12(CNC(C3C(=C)C3)=O)CC(SC)(C1)C1(CN(c3ccc(C(=O)OC)cn3)C1)O2 C1(C(N2CCC(C(N(CC(COC)O)C)=O)C2)=O)(OC)CCCCC1 N1(C(C(C=C)O)=O)CCCCC1C(=O)NC1(C(=O)NC(C)C)CC1 C1(CNC(c2c(C)sc(C)c2Br)c2n(CC)nnn2)CCC2(CCOCC2)CC1 N1(C(COCC(=C)C)=O)CC(N(C(=O)CCc2ccc(C)nc2)C)C(O)C1 C(C(C)(C)CC(=O)N1CCC(c2ccon2)C1)NC(C1C(OC)(OC)CC1)=O C=C(Cl)CCC(=O)NC1CCCC(CC(=O)NC2CCCC(CO)C2)C1.OC N1(C(CC(C=C)(C)O)=O)CC(C(=O)Nc2ccc(F)nc2C)CC(C)(C)C1 C(c1ccncc1)=CC(N1CCC(CNC(CN(C2CCSC2)C)=O)C1)=O C1(NC(C(C)C2CCC2)=O)CC(O)C1CC(=O)NCCCC(N)=O c1(CCC)cccc(C(=O)NCCC2CCN(C(=O)C=CSC)CC2)c1 CC1CC(O)CCN(C(C2CCC(O)CN2C(=O)COC2CCC2)=O)C1 c1(C(=O)NC(C)C(C)(C)NC(=O)CC2CCCCC23CC3)ccc2cnsc2c1 N1(C(C=CC(c2ccc(C)cc2)=O)=O)CC2OCC(NC(=O)C3=C(Cl)CC3)C2C1 C1(NC(C(C)SC(F)(F)F)=O)CCCCN(C(c2cocn2)=O)CC1 C1(C(=O)NCCNC(C2(CC)CC2)=O)CCCN(C(C2C=C2C)=O)C1 Cc1ccn2cc(CNc3cc(N(CC(F)(F)Br)C)nc(C)n3)nc2c1 N1(c2nccc(OC)n2)CCN(C)CC1CNC(c1cnn2cc[nH]c12)=O C(=O)(C(C(C)(C)C)c1ccc(C)cc1)N1CC(CNC(c2c(CC)ocn2)=O)C1 N1(C(C(C)C(C)(C)C)=O)CCC(F)(F)C(CNC(=O)CCCc2cc[nH]n2)C1 C1(CNC(c2cnc[nH]2)=O)CCN(C(=O)Cc2cc(Cl)cc(Cl)c2)C12CC2 Cc1ccc(Br)c(-c2nnc(NCCN3C(C)CCCC3C)o2)c1 CC(=O)CCC(=O)N1CCC(F)(C(=O)Nc2ccccc2SC(C)C)C1 C(=O)(C1=CCCCC1)NC1C(NC(=O)CCCN2CCCC2)COC1 C(C(C)(O)CNC(C1CCCN1C(c1cc[nH]c1)=O)=O)SC C1(C(=O)NCCCN(C(=O)C2=CCC2)C)CCN(C(=O)OC(C)(C)C)CCO1 N1(C(c2c(CC)nns2)=O)CCSCC1CCNC(=O)Cc1cnn(C)c1 Cc1nc(N2CCC(C(C)NC(=O)CC(C)C(C)C)CC2)ccc1C#N c1(CC(C)C(=O)NC(C2CCN(C(C3C(C)C3C)=O)CC2)C)ccc(O)cc1 N1(C(c2cc(C)n(C(C)C)n2)=O)CCC(C)N(C(=O)CC(O)C(C)(C)C)CC1 Cc1ccc(C(=O)NC2CCC(CC(=O)N(CCF)C3CC3)C2)cc1C#N C1(CCC)(NC(=O)C(C2CC2)SC)CCCN(C(=O)CN2CC(=O)NC2=O)C1 c1(CC)nc(-c2nc[nH]n2)sc1C(=O)N(CCNC(=O)C(F)F)CCOCCO C(=O)(CC(C)(C)C#N)N1CCCC(CCC(=O)N(CCCF)C)C1 c1(C(=O)NCC(CC)N(C(=O)C=CC2CCOCC2)C)cc(C)c(Cl)c(C)c1 c12cc(cc(Cl)c1F)OC(C)(C)CNC2=O.C(=O)(NOOC(F)F)OC(C)(C)C C1(C(=O)NCc2cccnn2)CC12CCN(C(=O)CC1COCC1O)CC2 CCC(CC)(CCNc1ncc(C)cn1)NC(C1CC2C=CC1CC2)=O N1(C(Cc2c(C)scc2)=O)CCCC(C(C)NC(=O)Cc2cncc(F)c2)C1 N1(C(c2cnc3c(c2)OCCN3)=O)CCCC(C2CCCN(c3nncs3)C2)C1 C(C(=O)NNc1ccccc1-c1nn[nH]n1)(C(C)C)N(C(C)(C)C)CC N1(CC2(C)CCN(Cc3cnn(C(C)(C)C)c3)CC2)CCc2ccsc2C1 C(C1(C)CCCc2ccccc21)NC(C=Cc1c(C)n(C)nc1)=O c1(NC(C)=O)cc(C(=O)NCCN(C(=O)C(O)CC(F)F)C)ccc1C N1(C(C2C(COC)CC2)=O)CC(CNC(=O)C(=CC2CCCCC2)F)CCC1C C(=O)(CC(CNC(=O)C(C)C#N)OC)NCCCSCC N1(C(CN(C(COC)=O)C)=O)CCC(C)C(NC(c2cc(Cl)ncc2OC)=O)C1 C1(C2CCOCC2)(C(N2CCC(N3CCN(c4nnco4)CC3)CC2)=O)CC1 N1(C(C=C(C)c2ccsc2)=O)CCC2(CCC2)C(NC(=O)CC2COCCO2)C1 C1(NC(C2(CC=C)CN(C(=O)Cc3cc(OC)no3)C2)=O)CCOCC1C c1(NC2CCCN(C(C3CCC(CC)O3)=O)C2)ncc(C(C)(C)C)cc1C#N c1(C(N(CCC(C(C)C)NC(C2(SC)CC2)=O)C)=O)ncc(C)cc1C c1(CC)nc(C)c(C(=O)N(CCC(C)(C)NC(c2cnc(C(C)=O)s2)=O)C)o1 c1(C(c2n(CC)nnn2)NC2CCCSCC2)c(F)cccc1Br c1(CC)cccc(CC)c1C(=O)NC1CN(C(=O)CCC2CCCOC2)CC1C C(=O)(CC1C(=O)N1)NC.C1(N2C(CNC(=O)OC(C)(C)C)CC2)CCCCC1 c1(C(N2CCN(CC(=O)N(C)C)CC2)=O)cc(Br)c(F)cc1Cl c1(C(N2CCC(CF)CC2)C(=O)NCCOCC)ccc(C(F)(F)F)c(Cl)c1 c1(CC)nn(C)c(CC)c1C(=O)NC(C)C(CO)NC(=O)C(N)=O c1(OC)cc(O)ccc1NC(=O)CC(C)(C)CNC(C1CCC(O)CN1C)=O C(CCN=C(NCC1OCC1(C)C)N1CCC(CC(C)(C)C)C1)OC(C)C c1(NC(C2(C)CCN(C(c3ccc(C#N)cc3Cl)=O)C2)=O)nc(Cl)c(Cl)cc1Cl c1(C(N2CC3C(CNC(C(=C(C)C4CC4)F)=O)C3C2)=O)coc2ccc(F)cc12 N1(C(c2cnn(C3CCCCC3)c2)C(=O)NCCCSC)CC(O)CC1C N1(C(CC)Cc2ccc(F)cc2)CCC(O)(C(=O)OCc2ccccc2Cl)CC1 c1(C(N2CC=CC(NC(C(C)(C3CC3)NC(C)=O)=O)C2)=O)cc(F)c(F)cc1O N1(C(C(C)C)=O)CCCCC1C1CCCN1C(C1CC2CCC(C1)N2C)=O c1(C(N2CCC(NC(COC(CC)(C)C)=O)CC2)=O)c(N)sc2c1CCSC2 N1(C(CC=C=C)=O)CC2CS(=O)(=O)CC2(CNC(=O)CCCN(C)C(C)C)C1 CC(C)(CNC(c1cc(Cl)n[nH]1)=O)CC1CN(C(=O)CCN2CCC2)C1 C1(NC(c2c(C)onc2CO)=O)COC2(C1)CN(C(=O)CC1(C)CC1)C2 Cc1cnc(C(=O)N(CCNC(=O)CCc2scnc2C)C(C)C)c(Br)c1 c1(C(=O)Nc2c(OC)cc(C(F)(F)F)cc2)cc2n[nH]cc2cc1-c1cnoc1 N1(C(C=Cc2ccc(C)nc2)=O)CCCC12CCN(C(=O)Cc1ncc(C)s1)C2 CCC(C)C(C)(O)CC(C12CCCC1C2(F)F)=O.C12C3CCN(CC13)NC2=O C(CCCCC(=O)NCC1CC(F)(CNC(C2CCCC2C)=O)C1)SC c1(C(=O)NCCC2CCN(C(c3c(O)cccc3Cl)=O)C2)cccc2occc12 C(=O)(CC(C)(O)C(F)(F)F)NC1CC(CNC(c2ccc(C)cc2)=O)CC1O CC(C)CC(C(=O)NC(C1CCOC1)C1CC1)ONC(=O)CC1CCCCC1O CC(CN(C(=O)CCC1CC1(F)F)C)C(=O)NCC(=O)NCC1CC1 C1(NC(CC(C)n2cccn2)=O)CN(C(c2cnns2)=O)CC2(CC2)C1 C1(C)(CNC(CCC2(C)CN(C(=O)CC#N)C2)=O)NC(=O)NC1=O C(C)(C)(CC(=O)N1CCCC1CCCNC(=O)C(C)Cc1cnc[nH]1)OC N1(C(C(C)OC)=O)CC2(CC(NC(=O)C(F)OC(F)(F)F)C2)C1 N1(C(C(C(CC)C)O)=O)CCn2c(nc(C(=O)NCC=Cc3ccco3)c2Cl)C1 N1(C(C(c2cccc(F)c2)C)=O)CC2=C(C1)CN(C(c1cc(Cl)nn1C)=O)C2 N1(C(c2cnn(C=C)c2N)=O)Cc2occ(C(=O)NC3CC4CC(O)C3C4)c2C1 C1(CCNC(CN(C)CCC2CCCC2)=O)CCCN1C(c1cncnc1)=O Cc1cc2nc(C(N3CC4CCC(N)(C4)C3)=O)[nH]c2cc1C Cc1cc(F)ccc1C(=O)NC1(C)CCCN(C(C2(C(F)(F)F)CC(O)C2)=O)C1 CC1(C)CC(=NO)c2cnc(NC(=O)COc3ccc4nccnc4c3)nc2C1 C(=O)(C1=NOC2COCC12)NCC(CC=C)NC(c1cn(C(C)C)nn1)=O C(=O)(C(C)(C)CS(C)(=O)=O)NC(C(CO)NC(c1n(CC)c(O)nc1)=O)C C1(C(=O)Nc2ccc(F)nc2)CCCC12CCN(Cc1cc(Cl)cc(Cl)c1Cl)C2 c1(C(=O)NCC(CCNC(=O)COC(F)F)OC)c(SC)cccc1F c1(C(N2CC(C(C)NC(=O)COC(F)F)OCC2)=O)c(F)cc(F)c(F)c1F C1(NC(c2cccc(NC(C)=O)c2)=O)CCN(C(C2(CN(C)C)CC2)=O)CC1F O=S(=O)(c1cccnc1N1CCCC(CC(F)F)C1)NC1CC2(C1)CC21CCC1 C(=O)(N=c1c(CS)c[nH]cc1C(F)(F)F)c1c(C)c(Br)ccc1F c1(C(=O)OC)ccc(CN2CC3(CN(C(C4(C)CCOCC4)=O)C3)C2)c(Br)c1 c1(C(N2C(C)CC(NC(=O)CCC3CC3(F)F)CC2)=O)nc2ncccn2n1 CC1C(NC(=O)Cc2ccccc2F)C(C)CCN1C(c1ccc(C#N)cc1)=O N1(C(C2CC(F)(F)CN2CCNCCO)=O)CCCC12CN(Cc1ncco1)C2 CC(C)(C)CC(CO)NC(C1COCC1NC(=O)CCC1OCCO1)=O CCCCCC(O)C(=O)N1CCC2C(C1)CN2C(=O)CP(C)(C)=O N12CCC(N(C)C)(CC1)C2.CC(C(=O)O)=CC(=O)N(C)C(C)C c1(C(=O)NCCNC(c2cc3ncccc3o2)=O)snc2ccccc12 c1(OCC(ONC(=N)Cc2ccccc2)=O)cc(Cl)c(Cl)cc1Cl c1(C(=O)NC(CCN(C)C(C2CCOC2=O)=O)C(C)(C)C)ccc2c(c1)CCO2 CC1CN(C(C2(CNC(=O)Cn3cccn3)CC=CC2)=O)CC(C)N1C c1(CNC(C2(NC(CCCOC)=O)CCSC2)=O)cc(O)cc(F)c1 c1(OC)ccc(OC)c(CCC(=O)NCCN(C(=O)CC(C)C)CC(C)O)c1 Cc1ccc(CC(=O)NC2CC(CC(=O)Nc3ncco3)C2)o1 C(CCCC(=O)NC1(C2CCCN2C(=O)CSc2nnc(S)s2)CC1)OC(C)C N1(C(CCSC)C)CC2COCC2(C(=O)N(C2CC2)Cc2ccc(C)cn2)C1 Cn1ccc2cc(S(=O)(=O)NCCCCCc3ccccc3)ccc12 c1(OC)ccc(C(C)C(N2CCC(NC(C3CC=CCO3)=O)CC2)=O)cc1OC c1(C(C)N(C(=O)C(=O)NC2CCCC23CCC3)C)ccc2ccccc2c1 Cc1ccccc1C(C)(C)C(N1CCC(F)(C(F)(F)F)C1)=O C1Cc2[nH]c(=NCCOC3CCOC3)nc(N3CCC(CF)CC3)c2C1 N1(C(C(CC)N(C)C(C23CC(F)(C2)C3)=O)=O)CC2CCC(O)C2C1 c1(C(=O)NC(C)CCN(C(=O)CC2(O)CCOC2)C)cc2n(n1)CCCC2 c1(C(N(C(C(=O)NCC2(CC=C)CCCC2)C)C2CC2)=O)sc(F)cc1C N1(C(C2(CC#C)CCN(C(=O)CC3CSC3)C2)=O)CCC(C(=O)NC)CC1C O=C(C1=COCCC1)NC(C1CCCC1)CNC(c1cscc1C1CC1)=O N1(C(CC(C(=C)C)OCC)=O)CC2(CCCC2NC(C2CCC(N=[N+]=[N-])C2)=O)C1 C1(NC(c2cc(CC)no2)=O)CCC(C)N(C(=O)Cc2csnc2C)C1 C1(CSC)CCCN1C(C1CCC(NC(=O)C=C(C)C2CC2)C1)=O Cc1ccc(OCCC(=O)N(C)CCNC(C2CCN2S(C)(=O)=O)=O)cc1C N1(C(CCC(=C)Br)=O)C2CCC1CN(C(c1c(C)n[nH]c1C)=O)C2 C1(C(=O)NC(c2ccc(Br)cc2)C(N)=O)CC(=O)c2ccccc2C1 C1(C)(CNC(c2c(OC)csc2)=O)CCN(C(C2(c3ccccc3Cl)CC2)=O)C1 Cc1cccc(CCC(=O)NC2CC(NC(=O)CC(C)(C)C)C2)c1Cl c1(C(=O)NC2CCCN(C(CCC=C=C)=O)CC2)cc(F)cc(F)c1N c1(C(CC(=O)NC2CC(CNC(CCOC)=O)OCC2)O)cc(Cl)cc(Cl)c1 C1(C(=O)NCC(CNC(C2(C#N)CCC2)=O)CO)CC2CCCCCC12 n1(CC)nc(Br)nc1C(N1CCOC(COC)C1)C(=O)NC1CC1.C1CC1 N1(C(c2ccnnc2)=O)CCC(CC#C)(C(N2CCN(C(=O)CCC)CC2)=O)C1 C1(NC(C2CC23CC(O)C3)=O)CCCCN(C(c2c[nH]nc2C(F)(F)F)=O)C1 c1(C(C(=O)O)NC(N2CCCC(C(=O)OC)C2)=O)ccc(F)cc1C c1(C(C)=O)ccc(C(=O)NCC(=O)Nc2cnn(CCN(C)C)c2)cn1 C(=O)(C(CC(C)C)C(C)C)N1CCC(NC(c2c(CC)occ2C)=O)C1C1CC1 N1(C(C2(C#C)CCC2)=O)CC2CN(C(c3cc(F)ccc3CC)=O)CC2C1 c1(C(=O)NC2C(C)CN(C(C3CCCC3O)=O)C2)cccc2nc[nH]c12 c1(C(=O)NC(CNC(C(Cc2c(C)cccc2)C)=O)(C)CO)csc([N+](=O)[O-])c1 C12(CNC(c3c(N)cccn3)=O)CCCC1CN(C(=O)CCc1cnc[nH]1)C2 N1(C(c2cnn3c2CCC3)C(=O)NCCSC)CCC2(CCCCN2C)C1 C1(NC(N2CCCCC2c2cccc(O)c2)=O)CCC12CCCO2 c1(OC)cc(CN=c2[nH]cc(CC(=O)NCCN(C)C)s2)cc(OC)c1O N1(C(CSC)=O)CCC(C2CCN(C(=O)COC(=O)Nc3ccc(F)cc3)C2)C1 c1(C(N(CCCN(C(CN(CC)CC)=O)C)C)=O)csc(C)c1CC Cc1ccc(CC(C)C(=O)NC2CCC(F)(CNC(C3(CCO)CC3)=O)C2)cc1 n1(CC)cccc1C(=O)N(CCCCN(C)C(C1(C)C=CCC1)=O)C C(=O)(C(O)C(C)(C)C)NC(C)CCCCNC(C1NC(=O)CC1C)=O C1(F)(C(N(C)CCOCC2CC2)=O)CCCN(C(C2(CO)CCCO2)=O)C1 c1(C(N2CC(C)(CNC(C(CCN(C)C)O)=O)OCC2)=O)c(F)ccc(F)c1F C1(CNC(C(CC2CC2)OC)=O)CC(C(F)(F)F)CN1C(=O)CCC1CC1 CCCCCCCCCC(=O)NCC1CCC1NC(=O)C(C)NC(C1CCC1)=O C(=O)(C(F)CC(C)(C)NC(C1CC1(C)C)=O)N1CC(CC(C)C)OCC1 c1(SC)cc(C(N2CC(F)(CNC(C3(N4CCOCC4)CC3)=O)C2)=O)ccc1N C(=O)(CCCCC(C)C)NCCCN(C(CC(N1CCC(CC)C1CC)=O)=O)C S(=O)(=O)(c1ccc(NC(=O)C(F)(F)F)cc1)N1CC(C)OC(C(N)=O)C1 N1(C(CN(CCC)C)=O)CCc2ccc(CNC(C3CCC(=O)N3)=O)cc2CC1 c1(C(=O)NC2CCCC2(F)F)ccc([N+](=O)[O-])cc1C CC1CCC(NC(C23CC(CC(F)F)(C2)C3)=O)CN1C(=O)CCn1cnnn1 C(=O)(CC(C)C(F)(F)F)N1CCCN(C(c2ccc(C(=O)OCC)cc2)=O)CC1 c1(C(N(CCCNC(=O)C=CCOC2CCOCC2)CC)=O)c(C)coc1C N1(C(C(C2CCCO2)NC(=O)C(c2ccccc2)F)=O)CCc2ccncc2C1 C1(OC)CC(CNC(=O)C(C2CCOCC2)O)N(C(=O)C=Cc2cc(C)no2)C1 N1(C(c2cccc(SC)c2)=O)CC2CCC1CN2C(C1CC(C)=NO1)=O c1(NC(C2C=CCN2C(=O)C=CCBr)=O)ccnc(F)c1 c1(CC)cn2c(n1)CC(C(=O)NC1C3CCCC1CC(N)C3)CC2 C1(NC(C(C)OCc2ccc(C)cc2)=O)C2CCC1N(C(=O)Cc1ccno1)C2 n1(CC)nc(C(=O)NCC2(F)CC(NC(C3CC(C(C)(C)C)C3)=O)C2)ccc1=O N1(C(C=C(C)Cl)=O)CC2CC(C1)N(c1nnc(-c3ccccc3)s1)C2 N1(C(CCC(=O)NC)=O)CC2(C(=O)NCC3CCC(C)(C)O3)CCC1CC2 N1(C(CCC)=O)CCC2C(C1)CN2C(C1CCCN1Cc1ccccc1)=O CCC(CC(=O)NCC1CN(c2ncc(C(C)(C)O)cn2)CCO1)CC(F)(F)F c1(C(C)C)nc(NCCc2cc[nH]n2)cc(=NCc2csc(Br)n2)[nH]1 N1(C(C(CC#C)O)=O)CC2CC(C1)CN(C(=O)C=C1CCOCC1)C2 C1(C(=O)NCc2c(C3(C)CC3)cccc2)CC(F)CN(Cc2ccc(Br)[nH]2)C1 C#Cc1cc2c(cc1-c1cn(-c3ccc4nc(CN(C)C)sc4c3)nn1)OCO2 N1(C(CCSCC(=O)OC)=O)CC(CNC(c2csc(C)c2C)=O)C(O)C1 c1(C(N2C(C)(CNC(C3(OC)CC3)=O)CCC2)=O)ccc(C)c(F)c1Br C(=O)(CC(C(F)F)NC(=O)C(C)=C1CCC1)N1CC(CCC)OCC1 C(C(C)(C)CC(=O)N(CCNC(=O)CC1CC(OC)C1(C)C)C(C)C)OC N1(C(CC2CC(=O)NC2)=O)CC2C(C(F)(F)F)CC2(NC(c2cnccn2)=O)C1 O(N=C(C(=O)OCC)C(=O)N1CCCC(c2c(C)nn(C)c2C)C1)CC c1(CC(=O)OCC(=O)NCc2ncc(C)s2)cccc(OC(F)(F)F)c1 C1(CNC(c2cnn(CC)n2)=O)(CO)CCCN1C(c1cn(CCO)nc1C)=O c1(CC)[nH]nc(C(N2CC3C(C(=O)NC(COC)CCO)C3C2)=O)c1C CCC(CC)CC(F)C(=O)NCC1COC(C)(C)CN1C(C1CC(C)(C)CO1)=O C1(NC(C2CC=C(C)CC2)=O)C2CC1CN(C(=O)CCOc1ccccc1F)C2 C1(C(=O)NC(C)(CNC(=O)CCc2ccncn2)C2CC2)CCCS1(=O)=O c1(C(N2CC3C(CNC(c4ccn(CC)c4C)=O)(C3)C2)=O)ccc(Br)cc1N Cc1cc(C(=O)NC2(CCNC(=O)CC3OCCC3(C)C)CC2)ccc1F C1(N(C(=O)C=Cc2ccoc2)C)CC2CCC(C1)N2C(C1CCC2CC12)=O C1(O)(CC)CN(C(=O)C(O)CNC(=O)CSCC(F)(F)F)C1 Cc1cc(=N)[nH]cc1C(=O)NCC1CC(F)(CNC(=O)CCc2cnc[nH]2)C1 C1(C(=O)NC2CCN(C(c3c(CC)nns3)=O)C2)COCC(C)(C)O1 c1(CCC(N2CCC(Cn3cc(C(C)(C)OC)nn3)C2)=O)ccc(Br)cc1F C1(C(=O)NCCn2c(CC)ncc2)CC(C)(C)CN1C(=O)C(COC)CC c1(CNC(=O)CN2CCCC2=O)ccc(C2(NC(CSCCOC)=O)CC2)cc1 c1(N2CC(C)(C)OC(CO)C2)nc2c(c(=NC3CC(F)(F)C3)[nH]1)CCCCCC2 CCC(C)(CNC(=O)C(C)C(F)F)C(=O)N1CC(n2ccnn2)C1 N1(C(=O)CCc2cnccn2)CC2(CCCN(C(C34CCCCC3C4)=O)C2)C1 c1(C(N2CC(NC(c3cnc[nH]3)=O)C3(C2)CC3)=O)c(F)cc(Br)cc1Cl N1(c2ccnc(C)n2)CCC2C(CCN2Cc2ccc3nc[nH]c3c2)C1 C1(C(=O)NCCC2(CNC(CCCOC)=O)CC2)(CCF)CCOCC1 c1(C(=O)NCC2CCC(NC(Cc3nc(CC)[nH]n3)=O)C2)nc(C2CC2)oc1C c1(C(=O)NCC2N(C)CCN(C(CCN(C)CC)=O)C2)ccc2[nH]nc(O)c2c1 N1(C(C(N2CCCNC2=O)C)=O)CC=C(CNC(C2CCCCC(=O)N2)=O)CC1 [N-]=[N+]=Nc1ccc(-c2cn(CCC(N3C4CCC3CC(O)C4)=O)nn2)cc1 N1(C(c2n(CC#C)cnn2)=O)CCC2CN(C(=O)C(CC)CCOC)CCC12 C1(CC)CN(CC)CCN1C(C1CCN(C(c2nocc2C(C)C)=O)CC1O)=O C1(N(C(c2c(C)scc2)=O)C)CCN(C(=O)CCCC(=O)NC(C)C)CC12CC2 C12(C(=O)NCCOCCN(C)C(c3csc4nnsc34)=O)CC(C1)S(=O)(=O)C2 N1(C(c2nc(C)cnc2C)C(=O)NCCSCC)CCC(C)C2(CCCCC2)C1 Cc1nc(CO)sc1C(N1CC(CNC(C2(C(F)F)CC(F)(F)C2)=O)C(C)C1)=O C(=O)(C1=CCCS1)N(C1CCN(C(C2CCCCC2n2cccn2)=O)C1)CC C(=O)(C(C)C(O)CC(C)C)N1CCCN(C(C2(COC)CCCCO2)=O)CC1 c1(OC)cc(F)c(I)cc1CNc1ccccc1CN(C1CCCC(O)C1)C=O C1(NC(c2c(OC)cc(O)nc2)=O)CCN(c2ncc(C)cc2OC)CC1(C)C C1(NC(CS(N)(=O)=O)=O)CCCCC12CCCN(C(C1(CC3CCC3)CC1)=O)C2 N1(C(c2nncc(OC)c2)=O)CC2(CC2)CC1CNC(C1(CO)CCC1)=O C(C)(C)(CC(F)C(=O)NCCC1CCCC(C)C1)NC(C(CSC)O)=O c1(NCCC(COC)C(C)C)ccc(S(=O)(=O)N2CC(C)=CC(C)C2)c(Br)c1 c1(NCC(N2CC(NC(c3cc(OC)ncc3)=O)C2)=O)nn(C)c(=O)n(C)c1=O Cc1nn(C2CC2)cc1C(=O)NCCCN(C(=O)CC1(N(C)C)CCC1)C N1(C(=O)Nc2ccc(C)cc2)CC2CN(C(=O)CN3CCCCC3=O)CC12 N1(C(CCC=CC)=O)CCC(NC(=O)CCc2ncc(C)[nH]2)C2(CCC2)C1 C(C)(C)(CC(=O)N1CCC(OC)CC1)N(C(=O)NCC(n1cccn1)C)C c1(C(=O)NC(C)CN(C(=O)C(C)(C)N(S(C)(=O)=O)C)C)nc2c(s1)COCC2 c1(NC)cnc(C(C2CCCC2)NC2CCN(C(=O)COCC(F)F)CC2)cn1 c1(CC(=O)NCC(C)NC(CSCC=C)=O)cc(F)cc2c1OCOC2 Cn1cc(Br)c(CC(=O)NC(C)(C)CNC(=O)CCCn2cnc(C#N)n2)n1 N1(C(=O)COC2CCCC2)CCC(O)C1C(N1CC2CC2(CO)C1)=O C1(C(=O)NCCN(C(=O)Cc2ccc(C)s2)CC)CCCN1C1CCCC1 N1(C(c2cn(CC)nc2C(F)(F)F)=O)CCCC2(C1)CN(C(C1(F)CC1)=O)C2 c1(-c2nc(C(CO)SCC)n(-c3cccc(COC)c3)n2)ccc(OC)c(F)c1 C1(C(=O)NC2C(C)COCC2)CC2CCC(C1)N2C(=O)C(C)(C)CC1CC1 N1(C(C(c2ccccc2F)(C)F)=O)C2CCC1C(NC(=O)Cc1ccc(Cl)s1)C2 CCCCC(O)CC(=O)N(CC(=O)N(C)CC1(C#N)CC1)CC(C)C N1(C(c2cnc(OCC)s2)=O)CCC2(CCN(C(=O)CN3CCNC(=O)C3)C2)C1 N1(C(C2C(C(C)=O)C2(F)F)=O)CCC(NC(C23CC4CC2C3C4O)=O)C(C)C1 N1(C(=O)NC(C)C)CCCC(C(=O)NCC(F)F)C1.C1(=O)C(=O)NC2CC2CN1 c1(CC)cc(C(N2CCCCCC2CNC(c2nc(C)n(C)n2)=O)=O)ccc1F N1(C(C(C(C)C)N(C)C)=O)CCC(C2CC2NC(=O)CC2CCOCC2)CC1 N1(C(c2c(CC)n[nH]c2)=O)CC2(CCC(NC(=O)CN(C)C)C2)C1 C=CCC(C)(O)C(=O)NCC1(COC)CCCN1C(=O)CC1CNC(=O)O1 N1(C(c2ccc(-c3cnco3)cc2)C(=O)NC(CC)C)CCn2ccnc2C1C O=C(C1OCCc2c(Br)cccc21)N1CC(CO)OC(CO)C1 C1(C(=O)NC(CC)CN2CCCC2)C2CCC(C2)C1NC(=O)C(C)(C)COC C(C(=O)N=c1ccn(CC2CC2)[nH]1)=CC1N(C(c2cnn(C(C)C)n2)=O)CCC1 c1(C(=O)NCCC2CCN(C(CCCCC=C)=O)C(C)C2)ccsc1S(C)(=O)=O N1(C(C(C)c2cccs2)=O)CC(NC(C2CC2c2ccsc2)=O)C2(CCC2)C1 c1(C(N2CCC(N(C(C(F)OC)=O)CCO)C2)=O)ccc(C(F)(F)F)c(C)c1 N1(C(CN(C)CC)=O)CC2CC1C2CNC(=O)C(C)(C)c1ccccn1 c1(C(N2CC(NC(Cc3cc(C)sc3)=O)C3(C2)CC3)=O)cc(F)cc(C)c1N C#Cc1cccc(NC(=O)C(C2(C)CC2)NC(=O)C(CC)CC=C)c1 N1(C(C(CCC)CCC)=O)CC2CCC1C1CN(C(=O)CCP(C)(C)=O)CC21 c1(CCNC(C)C)nc(CSCc2ccccc2)nn1-c1ccccc1 c1(C(N2CCCC3(C2)CN(C(C2C4COCC24)=O)C3)=O)ccc2c(c1)CCCN2 n1(C(C)C)ncc(C(N2CC(CNC(c3cnc(Cl)s3)=O)C2)=O)c1Cl C1(O)(CNC(C2CCCC(=O)O2)=O)CCCN(C(=O)CSc2nc[nH]n2)C1 Cc1cc(C(C)C(N2CC(NC(C3CC3c3cccnc3)=O)C(C)C2)=O)c(C)o1 CCC(C(=O)NCC1COCCN1C(=O)CCc1ccc(Cl)cc1)C(C)(F)F C(=O)(C1=CCCCC1C)NC(C(=O)NCC(COC)(C)C)c1cccs1 c1(C(CC(=O)N(CCNC(C2CC(C)(CC)C2)=O)C)C)ccc(F)cc1 c1(C(COCCNCCCOCC)(C)C)cccc(F)c1Br C1(CC(N2CCC(C)(CCC)C2)=O)N(C(=O)C(C2CC2)OCC)CCC1(C)C N1(C(C(c2cccc(C)c2)F)=O)CC(CNC(c2c(C)ncn2C)=O)CCC1C C1(NC(CC=CCC)=O)CCCC(NC(C)C(=O)Nc2cc(COC)oc2C)C1 C(=O)(C1=C(Cl)CCC1)N1CCCC(N(C(=O)CC=CC(C)(C)C)C)C1 C#CCC(C(=O)NCCn1ccnc1C)NC(c1ccc(OC)cc1)=O N1(C(CN2C(C)CCC2)=O)CC(=O)NC2CN(C(=O)CSC(F)F)CCC12 C(=O)(C(O)CN(C)C)NCC(CC)N(C(=O)C(C)NS(C)(=O)=O)C N(S(=O)(=O)N1CCCC1)C(c1nncn1C1CCCC1)=O N1(C(c2n(C)ccc2)=O)CC(CNC(C2(CC3CCC3)CC2)=O)OC2(CCC2)C1 CCCCCC(CC)C(=O)N(C(C)CCNC(=O)CC1CC(C)(C)C1)C N1(C(c2cc(C3CC3)no2)C(=O)NC2CCCC2)C2CCC1CC1(C2)N=N1 N1(C(C2NC(=O)OCC2)=O)CCN(C(C2CC2c2ccccn2)=O)CC2(CC2)C1 C(C(CC(=O)NC(C(C)SC(C)C)=O)C1CCC1)N(CCCCO)C(N)=O c1(C(=O)NCC2CN(C(C=C(CC)C)=O)C3C2C3)cc2ncccc2s1 c1(NCC2(C=C)CCC2)cc(NCC(c2ccccc2F)OC)ncn1 C(CC(=O)N(CC(C)C)CCO)N(C(C1C(C(=O)OC)C1)=O)C1CC1 C1(OC)CCCCC1C(=O)NCCCN(C(=O)Cc1cscn1)C1CC1 N1(COC)CCCC(C)C1.c12noc(n1)C1CC1c1noc(n1)C21CC1 CCC(C)CCC(O)CC(=O)NCCOCCNC(=O)C=CC1CCC(C)CC1 C(C(Cc1ccc(Cl)cc1)C(=O)NC(CNC(=O)C=C1CCC1)C(C)(C)C)OC C(c1ccccc1)=CC(C(=O)NCC1(NC(COC)=O)CCC1)C N1(C(C2(CC#C)CCOC2)=O)CC2CN(C(=O)Cc3cscn3)CC(F)(F)C2C1 N1(C(C2C(C)=C2)=O)CCC(C)(C)C(CNC(=O)Cn2nc(C)c(Cl)c2C)C1 C(CCS(N)(=O)=O)c1cn(C(CNC(C2C(OC)CC2)=O)C)nn1 C(=O)(C1=NOC2(CCOC2)C1)N1CCN(C(CC(C)(C)C#N)=O)C(C2CC2)C1 C1(COC2CN(C(=O)C3CC3)C2)(NC(=O)Cn2cnc(C(F)(F)F)c2)CCOC1 C1(C(=O)NCc2c(C)nns2)CC2(CCN1C(=O)C#CC(C)(C)O)CC2 CCC(C(=O)NC(C)C(C)(C)NC(=O)C=CCF)NC(=O)CSC(F)(F)F N1(C(COC)=O)CCOCC(CNC(c2ccc(-c3nnc(O)n3C)cc2)=O)C1 C1(CC(N2CC(N(C(CN(C(=O)NC)C3CC3)=O)C)C2)=O)CC(O)C12CCC2 C12CC(F)(F)CN1C(=O)CO2.N1(C(C2C(CCC)C2)=O)CC(OCCSC)C1 c1(OC)c(C(=O)NCC(CNC(=O)CCC2CC2)OC)sc(C)c1Br C1(NC(c2ccc(CC)s2)=O)CC2CCC(C1F)N2C(C1COCCC1(F)F)=O C(CC(C)C)(C(=O)N1CCOC(CC(=O)Nc2cc(Br)cnc2C)C1)NC(C)=O c1(CC2(N)N(Cc3c(-c4nnc(C)o4)cccc3)CCCC2)ccc(Cl)c(Cl)c1 c1(OCC)c(C(=O)NC2CCC(NC(c3ccnc(C)c3N)=O)C2)cccc1F C(=O)(N=c1ccn(C)[nH]1)C1CN(Cc2c(OC)nccc2I)CC1O N1(Cc2c(C)n(C3CCC3)nc2)CCCc2oc(Br)cc2C1 N1(C(c2cscc2C(F)F)=O)CCC2(CCN(C(c3cccnc3F)=O)C2)C1 Cc1cc2nc(NCCc3ocnc3CNC(=O)C(C)N3CCC3)cc(=O)n2o1 C1(NC(C2C(C)CC2)=O)CC2CCC1N(C(=O)CCNC(N)=O)C2 C1(C(=O)NC(C)CNC(C2(N3CCOCC3=O)CC2)=O)Cc2ccccc2C1 C1(NC(C=CCCC)=O)CC2CCC(C1C)N2C(c1cncc(C(N)=O)c1)=O C1(NC(C(CC)CN(C)C)=O)CCN(C(=O)COc2ccon2)C12CCC2 Cc1cccc(OCC(=O)NC2CN(C(=O)CN3CCC3C)CC2F)c1C c1(C(=O)NCC=C)ccc(C(=O)NCC2CC2NC(c2cnc(Cl)cn2)=O)cc1 c1(OC)cccc2c1C(=O)N2.c1(C(CC(=O)NC)O)cccc(F)c1Br Nc1ccc(Cl)cc1C(N1CCCCC(NC(c2cnn3c2OCC3)=O)C1)=O c1(C(=O)NC23CC(NC(CCCCCOCC)=O)(C2)C3)cc(F)c(N)c(F)c1 c1(C(N2C(C)CC(NC(C3CCCCCC3)=O)C2)=O)cnc(Br)c(N)n1 C(=O)(CCCNC(c1c[nH]nc1C(F)F)=O)N(C)CC1CCCO1 CC(CC#N)C(=O)N1CCCC(CC(N2CC(C)C2)=O)C1.N(C)(C)C(=O)O C1(NC(Cc2c(C)cco2)=O)CC(NC(C2(C)CC2C)=O)C(O)C1 C(c1cccc(Cl)c1)=CC(=O)NC(CC(C)C)CNC(C1(F)CCOCC1)=O C1(C(N2CC(O)(C(C(=O)NC(c3nccs3)CC)F)C2)=O)CCC(C)(O)CC1 C(=O)(CS(=O)(=O)C1CCCC1)N1CCC(CC=C)(NC(=O)C(C)CCO)C1 c1(OC(C)=O)ccc(CNCc2cccc(OC3CCCC3)c2)nc1.N12CC(C1)C2 C1(C(=O)NCCN2C(=O)CNC2=O)CC2CN(C(c3n[nH]c4c3COC4)=O)CC2C1 C(=O)(CS(=O)c1ccc([N+](=O)[O-])cc1)NC1C2(CN(C(C(F)=CCC)=O)C2)CC1 N1(C(CC2N(C(C3C(C)C3)=O)CCC2)=O)CCOC(C)(C2CC2)C1 C1(NC(Cn2cc(CN(C)C)nn2)=O)CCCCC1CNC(C1CCN(C)C1)=O N1(C(C2C(C)C2)=O)CCOC(C)(CNC(C2CCN(CC(F)(F)F)C2)=O)C1 C=CC1(C(N2CC(CCO)C2)=O)CCN(C(=O)CCCCCF)C1 C=C(C)C(C)(O)C(=O)N1CCC1CNC(c1ccccc1N(CC)CC)=O c1(C(=O)NC(CCNC(c2ncn(C(C)C)c2)=O)C)nccnc1C(N)=O C(CC(CC)(CC)NC(c1cc(C)ncn1)=O)NC(CN(C1CC1)CC)=O c1(N(C(C2CCN(C(C)=O)C2)=O)CC2CCC(CC)O2)ccc(OC(F)(F)F)cn1 c1(C(N)=O)c[nH]c(C(=O)NC2CC(CCNC(C3(C4CC4)CCCO3)=O)C2)c1 C(CCC)(C(=O)NC(C)(CNC(=O)CC1CCCN1C(C)=O)CO)=CCC c1(CC)nn2c(=O)cc(CN(c3ccc(C)c(F)c3)C)nc2s1 c1(CN(Cc2ccc(CCC)s2)CC2(C)CCCC2)cccc(Br)c1 C#Cc1ccc(C(N2CCC(NC(=O)C(F)(F)C3(OC)CCC3)C23CC3)=O)cc1 C(C(CC(=O)NCC(CO)NC(C1CN2CCN1CC2)=O)C(F)F)N(C)C C(=O)(C(F)CC1CCCCC1)N(C(C1(CNC(C2(CC)CCC2)=O)CC1)C)CC N#Cc1ccsc1C(N1CCOC(C(N2CC(N3CCC3)C2)=O)C1)=O c1(C(=O)NCCCCN(CC)CC)c(CNC(C2CC2C2CCCO2)=O)nnn1C C1(NC(c2n(C)nnn2)c2cnc(Cl)s2)C2CCC(F)(F)C12 C1(COCc2cn(C3CN(C(C(C)NC(C)=O)=O)C3)nn2)CC(=O)C12CCCC2 C1(NC(CNC(C)=O)=O)CN(C(C2(Cc3ccccc3)CCOC2)=O)CC1N=[N+]=[N-] C=CCCCC(C)(C)C(=O)NC(CNC(c1cc(O)ncn1)=O)CO C1(CC)(NC(=O)CCn2cccn2)CCN(C(=O)CCc2ccc(Cl)cc2)CC1 C(=O)(C1=CCC(F)(F)CC1)NC1CCCC(NC(=O)C(=Cc2c[nH]cn2)F)C1 C1(CNC(C2(C)CN(C)C(=O)C2)=O)CCN(C(c2sccc2F)=O)C12CCC2 c1(CNC(=NC)NCC2(c3ccccc3)CC2(F)F)cc(C)ccc1Br C12(CNC(C3C(C#N)C3)=O)CN(C(c3cc(C(N)=O)no3)=O)CC1CCO2 C(CN=C(NCc1noc(C)n1)NCC1CCSC1)OC C1(CNC(CC2CC(OC)C2)=O)CC(F)(CNC(=O)CSc2n[nH]c(C)n2)C1 CCC(CC(=O)NC1C=CCN(C(C2(C)CCCO2)=O)C1)OC CCC(C)CCCCC(=O)N1CCC(C)(NC(c2cc(C#N)c(C)cn2)=O)CC1 N1(C(C(c2ccccc2)OC(C)C)=O)CCCN(C(C2CCCOC2)=O)C(C)C1 CCCC(C(=O)NCCC(=O)NCCN1CCCCC1)NC(=O)CC C1(N(CC)CC)CCN(C2c3ccn(n3)CCNC2=O)C1.C(CSC)SC C(=O)(CC(C(F)F)NC(=O)CC1CCC(=O)C1)NC(c1nc(C)[nH]n1)(C)C CC1(C)CC(=O)N(CC(N2CCC3(NC(c4cnc(N(C)C)o4)=O)CC3C2)=O)O1 CCC(C(=O)NC1CCCC1(C)CN(C(=O)COC1CCCC1)C)C(C)(F)F CCCCCCCCC(=O)Nc1cccc(F)c1I CC(C)C(O)(C(=O)N1CCN(C(=O)Cc2cnsc2)CC(O)C1)C(F)(F)F C1(SC)CCC(N=c2[nH]c3c(c(=NCCc4ccc(F)cc4)[nH]2)SCC3)C1 C(C(C)(C)C(=C)C)N(C(=O)Cc1ccsc1)CC#C.C1=CC=CCN(CC)C1=O c1(C(N(C2CN(C(c3c(C)onc3O)=O)C2)C)=O)cc(Cl)c(Cl)cc1N N1(C(CNS(CCCC)(=O)=O)=O)CCC(NC(=O)CCC2CCOC2)CC1C c1(NC(Cn2nnc(C)n2)=O)cnc(C)c(C(=O)N(C)C)c1 c1(C(C)C)ccc(F)c(C(=O)NC(C)CN(C(=O)COc2ccc(F)nc2)C)c1 C(CC(C(=O)NCCc1cc(C)no1)NC(C1CCN1CC)=O)OCC N1(C(c2ccc(C)nn2)=O)CCC(CNC(=O)CC2(C)CCOC2)CC1C Cn1c(C(N2CC(NC(c3occc3F)=O)C(C3CC3)C2)=O)cnc1[N+](=O)[O-] CCC(C)CCCCC(=O)NCC(CC(=O)NCCC(C)C)C1CCC1 C=CCC(CC(C)C)C(=O)N(C)CCN(C(=O)CN1CC(=O)NC1=O)C(C)C C1(OC)CCC(C)N(C(C2CCCN(c3nccnc3F)C2)=O)C1 C(C(CNC(c1ncnn1CC)=O)C(F)(F)F)NC(CCCC#C)=O C=C1CCN(C(C2CCC(=O)C2)=O)C(C(=O)N(C)CC2(COC)CCC2)C1 C1(CNC(C)=O)CCCN(C(=O)NCc2cccc(Br)n2)C1 C1(NC(c2c(C)nc(CC)s2)=O)CC2(NC(C3CCN(C)C3=O)=O)COC1C2 N1(C(C2CC(C)N2C(c2ccc(CO)o2)=O)=O)CCCCN(C)CC1 C1(C(C)C)C(NC(=O)CCCC2CCCC2)CCN1C(c1cnc(C2CC2)o1)=O N(C(=NCCCCl)NCc1c(C)cccc1F)C1CC(OC)C12CCC2 N=c1[nH]nc(C(N2CC(CC(F)C(=O)NCC3CSC3)C2)=O)[nH]1 S(=O)(=O)(c1ccccc1)NC(=O)CC(=O)NC(c1ccc(O)cc1)C(=O)O c1(C(=O)NC23CC(NC(c4cnc(O)s4)=O)C(OC2)C3)n[nH]c2c1CCCC2 Cn1cc(CC(=O)NCC2CCC2NC(=O)COC2CCOCC2)nn1 Cn1nnc(C(N2CCC(C)(CCNC(C3CCC3C(F)F)=O)C2)=O)c1N Cc1ccc(C2(NC(=O)C(C)(Cc3nn[nH]n3)c3ccccc3)CC2)cc1C Cc1ccc(NC(N(C2CCC2)CC2CCCCC2C(C)(C)C)=O)c(C)c1 c1(C(C)NC(=O)NCCC2(CC(=O)OCC)CC2(F)F)ccc(C)cc1 C1(NC(c2c(C)nc(CC)o2)=O)CN(C(=O)COc2cccc(F)c2)CCC1F n1(-c2cccc(C(=O)OC)c2)cc(C#CCNC(C)=O)nn1.C12(CC1)N(C)C2 CC1=C(CNC(=O)CCC2CCCN(C(c3cc(C)c(C)s3)=O)C2)COCC1 c1(OC)ccc2nc(CNC3(N)CC4CCC(C4)C3)[nH]c2c1 N1(C(C2CCC2)=O)CC2CCC(C1)N2S(=O)(=O)CCC(F)(F)F.C1(C)CCC1 c1(NC(Cc2ccc(-c3n(C)cnc3)c(F)c2)=O)cc(F)c(F)c(F)c1F N1(C(c2cn(C)[nH]c2=N)=O)CC2CCCCCC2C1 C(=O)(CC1=CCN(C(=O)CC2OCCO2)CC1)NCC1N(CC)CCCC1 C1(C(C)C)C(=O)N1.N1(C(CCOCCSCC)=O)CCC(C)C1CC N1(C(CCC(=C)Cl)=O)CCC(F)(F)C(CNC(C2CCN(CC)C2)=O)C1 N1(C(c2snc(OC)c2Cl)C(=O)NC(CC)C)CCC2(CCCO2)C1 CCCCCC(C)CC(=O)N1CCC(CCC(N2CC3C(C)C3C2)=O)CC1 C(=O)(C1CC(O)c2ccccc21)N1CC(C)(NC(c2csnn2)=O)C1 CC1=C(C(=O)NC2CCC(CCNC(=O)Cc3ccno3)C2)COCC1 C1(CNC(c2nc(C)oc2)=O)CC2(CCC2)CN1C(=O)C(C)Oc1ccccc1 c1(OCC(C)NCC(O)CN(C(=O)CCCN2CCCC2)C)ccccn1 C1(NC(Cc2ccc(C)nc2)=O)CC2CC(C1)N(C(C1(C)CCOC1)=O)C2 C12CON(C(=O)c3ccnc(c3)S1)C2.C1(C(=O)N(C)C)CCCN1OC c1(C(=O)NCC2C3CN(C(CS(C)(=O)=O)=O)CC32)c(N)sc2c1CCC2 N1(C(C(COC)(C)C)=O)CCC2(COC(CNC(c3conc3C(C)C)=O)C2)C1 c1(C(N(CCc2ccc(OC)cc2)C)=O)cc2c(Br)ccc(C=O)c2[nH]1 C=CCC(C)(C)C(=O)N1CC(CO)(NC(=O)C(CC(=C)C)OC)C1 C1(NC(C(C)Sc2nncn2C)=O)CCN(C(c2ncn(C)n2)=O)C12CCC2 CN1CC2(CN(C(=O)C(c3ccoc3)NC(=O)CNc3ccccn3)C2)C1 c1(NC(C2CN(CCC=C)CC2C)=O)nc(-c2ccccc2)c(C)c(C)n1 c1(C(=O)NC(CCOC)CNC(c2cccc(OC)n2)=O)ccc2n[nH]cc2c1C O(N1C(=O)c2ccccc2C1=O)CC(=O)NC(C)C(CO)NC(=O)CNC(N)=O c1(C(=O)NC2CC(C)N(C(=O)CCc3nc(O)n[nH]3)C2)cnc(Br)c(N)c1 c1(C(=O)N=c2cc(CCO)[nH][nH]2)ccc2c(c1)CN(C(C1CC1C1CC1)=O)CC2 N1(C(C2CC(OC)C2)=O)C(CC(=O)NC2CC23CCCC3)C2CCCC12 Cc1ccc(C(N2CCCN(C(=O)C(C)CC(C)C)CC2C)=O)c(O)c1C C(=O)(C(CC(C)C)C(C)C)NC(C(=O)NCCCC(=O)OC)CCC1CCC1 C1(OC)CN(C(c2nccn2C)=O)C(C)(CNC(=O)CO)C1 c1(C(=O)NCC(C)NC(C2CCCN2CC(F)(F)F)=O)cc(F)ccc1F c1(C(=O)OC)sc(I)cc1NC(=O)CC1CN(Cc2c[nH]c(Br)c2)C1 Cc1ccc2[nH]c(C(=O)NCC3CCC3NC(c3ccncc3)=O)c(C)c2c1 C1(CC(=O)NC(COC)C(=O)OC)CN(C(=O)Cc2cn[nH]c2)CCC1C c1(C(=O)NC(CCCC)CNC(=O)Cc2csc(Cl)n2)cc(C)nc2ncnn12 c1(CNC(C2(CCN(CCC=C(Cl)Cl)C)CC2)=O)cccnc1 C1(CNC(CCC(C)(C)OC)=O)CCC2(CCC2)C1NC(c1nnccc1C)=O Cc1cc(C(=O)NC2CC(CNC(C3CC=CCO3)=O)C2)ncc1S(N)(=O)=O C1(NC(=O)CC2(NC(=O)CC3CC3)CC2)CCCC(CO)CC1 N1(C(c2ccncc2Cl)=O)CC2CCN(Cc3c[nH]c(Br)c3)C2C1 c1(C(N(C2CCN(C(C3CC3C(F)F)=O)CC2)CC)=O)c(Cl)nc2ccccn12 C(=O)(CC(O)CCNC(=O)C(F)(F)C(C)O)NCCCN(CCCOC)C C(=O)(CC(C)(C)C(=O)N1CC2C(CC(=O)NCC(F)CO)C2C1)OC O=C(C1=CCCN(C(=O)CC2CCCO2)C1)NCC1CC(CF)C1 C1(CC#C)(C(=O)NCCN2CCCC(O)C2)CCN(C(=O)CCC2CC2C)C1 c1(C(C(=O)N(C2CCCN(C(c3cnnn3CC)=O)C2)CC)C)cccc(Cl)c1 C(=O)(C(CCOC(C)(C)C)NC(=O)On1ncc(C(C(=O)OCC)F)c1)OCC Cc1ccc(C(=O)NC(C)CC(C)NC(c2ccc(-c3cccs3)o2)=O)s1 N1(C(c2ccc(CCC)cc2)=O)CCN(C(=O)C(O)CF)CC(O)C1 N1(C(c2ccc(C(=O)OC)o2)C(=O)OC)CCC(n2cc(C(N)=O)nn2)CC1 c1(OCC)ccc(C)cc1NC(C1CC(NC(C2CCCCO2)=O)C1)=O C1(CNC(CNS(CC)(=O)=O)=O)CC(C)N(C(=O)CC2OCCO2)C1 N(C1CCCc2ccc(Cl)cc21)C(c1cc(C)c(C)s1)c1nnnn1C Cc1ccc(CCC(=O)N2CC(n3cc(CNc4nnc(C)n4C)nn3)C2)cc1 CCC(CC(=O)N1CCOCC1C(=O)NC1CC(F)(F)C1)C(C)(C)C CCC(C)CCC(=O)NC1CC(C)N(C(c2ccc(OC)nc2)=O)C1 c1(CNC(=O)CCC2CC(C(=O)NC3CC4CCCC4C3)C2)cccc2cc[nH]c12 C1(NC(c2c[nH]c(=S)cn2)=O)CCCCC1C(=O)NCC1CCCOCC1 C1(NC(C(C)NC(N)=O)=O)CCCCC12CCCN(C(=O)C(F)C(F)(F)F)C2 c1(C(N(C(c2ccc(S(C)=O)cc2)C)C)=O)ccnc2ncnn12 c1(OC)ccnc(C(=O)NCC2CN(C(=O)C(C)(C)c3ccsc3)CC2C)c1O C1(C(=O)NC2C(C=C)CN(C(=O)CC(C)(C)OC)C2)CCc2cnnn2C1 C=CCC(C)C(=O)NC1CN(C(=O)CSCC(=O)OC)CC1F C1(C(N)=O)CCCCC1C(=O)NC1CC(CNC(c2n[nH]cc2Cl)=O)C1 c1(C(N(CC(CC)NC(c2ccn(C(C)C)n2)=O)C)=O)ccc2snnc2c1 C1(C2(NC(C(C)CC3CCC3)=O)CC2)COCCN1C(=O)COCc1nc[nH]n1 CC1=CCCN(C(c2cccc(CN(S(C)(=O)=O)C)c2)=O)C1 Cn1nc(C(=O)NC2CC(C)(CNC(C3(C4CCCO4)CC3)=O)C2)c2c1CCC2 c1(OCC)ccnc(NNC(=O)c2cc(=O)c3ccccc3[nH]2)n1 c1(NC(C)=O)ccccc1CC(=O)NC1CC1NC(=O)CC1CC2C=CC1C2 c1(NC)ccccc1C(N1CC2CC2(CNC(=O)C2=CCCC2)C1)=O CC(C)(CNC(=O)CC1COCCN1C(=O)Cc1ccccn1)C1=CCCC1 c1(C(N2CCC(O)(C(=O)Nc3cc(Cl)c(Cl)cc3F)C2)=O)ccc(Br)c(Cl)c1Cl C1(NC(C2CC(CC)(CC)C2)=O)CCCCC1NC(c1cc(C)no1)=O C(CC(CNC(C1COCCO1)=O)NC(=O)COCc1ncnn1C)OC N1(CC)CCCC1C1CCCN1C(=O)Nc1ncccc1Cl N1(C(C)=O)CCC(C(F)C(=O)NCCCCN2CCCC2)C1 C1(CNC(C(CC)OCC)=O)CN(C(=O)Cc2cnn(C(C)(C)C)c2)CC(C)O1 C1(CNC(c2nnn(C)n2)=O)C2CN(C(c3cc(O)ncn3)=O)CC12 C1(C(C)(C)NC(C(C)(F)F)=O)CCN(C(c2ocnc2C2CC2)=O)CC1 N1(C(C)C)N=C(C(=O)NC2CC23CCN(C(C2CC2C#N)=O)CC3)CCC1=O CCC(CC)C(C)C(=O)NCC1(COC)CN(C(c2cnc(C(C)C)[nH]2)=O)C1 C1(CNC(C=CC2N(C(CCOCC#C)=O)CCC2)=O)CN2CCC1CC2 C1(CNC(CCSCCC)=O)CN(C(C2(N3CCCC3)CCC2)=O)CC1(C)C C1(C(N2CC(O)(CC(=O)NCCOCC(F)F)C2)=O)(OC)CCCOC1 c1(C(=O)NC2CCCC(NC(c3c(OC)ccs3)=O)C2)cc(Br)cnc1O c1(C(N2CC(C(C)NC(c3cc[nH]c3)=O)OCC2)=O)ccc2c(c1F)CCC2 Cc1cc(C(N2CCC(CCNC(=O)Cc3cnns3)C2)=O)nc(N(C)C)n1 CCC(CC(=O)N1CC(C(C)(C)O)(CNC(=O)C(C(C)C)NC(C)=O)C1)SC N1(C(c2ccnn(C)c2=O)=O)CC2CN(C(C34CCCCN3CCC4)=O)CC2C1 c1(C(N2C(C(N(C3CCC3)C)=O)C=CCC2)=O)c[nH]c2cnccc12 c1(OC)cccc(C(=O)N(C(c2ccccc2)CNC(=O)C(C)N(C)C)C)c1C c1(CC(=O)NCCC2CN(C(C3CCC(C#N)C3)=O)C2)ccc(O)c(F)c1 C(c1cccnc1C)=CC(=O)NCCNC(c1n(CC)ccn1)=O Cn1ncc2c(NCc3ccncc3)nc(N3CCC(C4CCCO4)CC3)nc12 C1(CC(=O)N(C(CN(C(Cc2nc(C)sc2)=O)C)C)C)CCCCN1C N1(C(C2C(C(C)C)CCC2)=O)CC(NC(C2CC(F)CN2C)=O)CC(O)C1 C1(C)(CNC(CN(CCC#C)C)=O)CCN(C(=O)C=Cc2cc[nH]n2)C1 c1(C(N(C(CC)CC)CC)=O)cc2cc(C(=O)O)ccc2o1 C(=O)(C(C(C)(C)C)n1cc(C(c2cccnc2F)=O)nn1)NCc1cc(C)c(C)o1 C1(C(=O)NC2(CSC)CCC2)CN(C(=O)C2=NOC(C)C2)CCN1C c1(NC(=O)NC(c2ccc(C)cc2)C=C)ccc(OC2CCC2)cc1 N(C(=NCCCSC)NCC1CCCC(F)C1)CC(=C)C C1(NC(CC(CC)OC)=O)CN(C(C2(C3CCC3)CC2)=O)CC(C)(C)C1 C1(C(=O)NCC(N2CCCC2CC(=O)NC2CCSC2)=O)C2CC3C(C2)C13 c1(C(C(=O)NCC(CCOC)NC(=O)C(C2CCCC2)OC)C)ccc(F)cc1 C(N=c1[nH]ncs1)C1CCN(C(C(=O)NC(C)C)=O)C1 CCCCC(F)(F)C(=O)NC1COCCN(C(c2ncccc2O)=O)C1 C(Cc1ccccc1)(C(=O)N1CCCC1C(C)(C)CNC(=O)CC1CC1)N(C)C Nc1cccc(C(=O)NC2(CNC(c3cncc(OCC(F)F)c3)=O)CCC2)c1 C(CC1CC1)(CC(=O)NCCCC1CCCC1O)NC(c1c(CC)nn[nH]1)=O C1(C(=O)NC2CN(C(c3cnns3)=O)CC2CO)CC12CCCCC2 NC(=O)CCCC(=O)NC1CC2CC(NC(c3ccc(OC(F)F)nc3)=O)C1C2 c1(C(N(CCCCCNC(C(CC)C)=O)C)=O)ccc([N+](=O)[O-])cc1C(F)(F)F CCCC(O)C(=O)NC(C)CCNC(=O)Cc1csc(Br)c1 Cc1cc(=O)c(C(=O)NC2(CNC(C3CCOC3=O)=O)CCCCCC2)cn1C C12(CC(N3CCC(O)C(CO)C3)=O)CCC1CN(C(c1n[nH]c(O)n1)=O)C2 c1(OC)cncc(C=CC(=O)NCC(c2ccccc2C)NC(=O)CC2CC2)c1 c1(COC)nn(C)c(Cl)c1C(=O)NCC(CO)NC(=O)C(C)n1cnnn1 C1(C)(C(N2CC=CC(NC(C(C(C)C)O)=O)C2)=O)CCCNC1=O C(CCN(C(=O)C=CCn1cncn1)C)(C(C)C)NC(C1(SC)CC1)=O N12CC3C(C3C1)CNC2=O.c1(C2(NC(c3cnccn3)=O)CC2)ccc(F)cc1 CCC(C)CC(C)N(C(=O)CC1CC(O)CN1C(=O)CN(C1CCC1)C)C CC(C)CCC(=O)C(=O)N1CC(C(N)=O)(CNC(=O)Cc2ccsc2Cl)C1 C1(CC)CN(C(c2cc(Br)ccc2Cl)=O)CCN1C(=O)C(C)CF N1(C(C2N(C(c3nc(CC)sc3)=O)C(CC)CC2)=O)CCN(C2CC2)C(=O)C1 c1(C(N2C(C(=O)NC3CCC4CC3C4(C)C)CC(C)C2)=O)cc2cccnc2[nH]1 C#Cc1ccc(C(=O)NCCSCC(=O)NC2CC(C3CCC3)C2)cn1 N1(C(C2(C)N(C(c3n(C)nc(C)c3F)=O)CCC2)=O)CC2CCCCC2C1 N1(C(C(C)OC)=O)CCN(C)CC1CNC(=O)CC1(O)CCCOC1 N1(C(c2ccn(CC)n2)=O)CCCC(C)C1CCNC(=O)CCc1cccnc1 c1(C2(C(N3C(CNC(=O)C=CC4CCC4)CC3)=O)CC2)ccccc1 C1(C(N2CCCC2Cn2cc(C3(O)CSC3)nn2)=O)CC2C=CC1C2 c1(C(N2CC(COC)(CNC(C3(C)CCCC3C)=O)C2)=O)cc(F)cnc1O C1(CCNC(c2ccc(C)nc2)=O)CCN(C(=O)Cc2cccc(Cl)c2)C(C)C1 c1(CCC)c(C(=O)NCC(C)(C)CCNC(=O)CC2CC3C=CC2C3)nnn1C N1(C(CC(CC)O)=O)CCC(O)(C(C)NC(=O)C(C)OCCN(C)C)CC1 c1(C(N2CC3N(C(C#CC(C)C)=O)CC(C3)C2)=O)n[nH]c2c1C(=O)CCC2 c1(OC)ccc(C(=O)OC2CN(c3ccnc(SC4CCOC4=O)n3)C2)cc1 CC(C)CC(C)(O)C(=O)N1CC(C(=O)NC(c2cscn2)CO)C(F)(F)C1 c1(C(N2C3CN(C(CCS(=O)(=O)N(C)C)=O)C(C3)C2)=O)cc2c(nc1O)CCC2 C1(N(C)C(=O)NC2CCOC2(C)C)COC(C)(C)OC1 C(=O)(C(F)CC(C)(C)C)N(CC(=O)NC1(CC=C)CCOC1)CCC Cc1cnn2cc(C(=O)NC(C)(CNC(c3ncncc3Cl)=O)C3CC3)cnc12 N1(C(C(CC(C)C)C)=O)CCN(C(c2cn(C(C)(C)C)cn2)=O)CC(CO)C1 C1(NC(CN(CCOC)C)=O)CCN(C(=O)Cn2nc(C)n(C)c2=O)CC1(C)C C(=O)(CC(C(=O)N1CCC(C)C1CNC(=O)CC1CC(O)C12CCC2)N(C)C)OC CC1(C)CC(NC(=O)CCN2CCC2)CN(C(=O)CCCCCNC(N)=O)C1 Cc1cc(NC(C2CCC3(CC3)N2C(=O)CSC(F)F)=O)c(C)c(C)c1 C1(C)(C(=O)NCC(=CC(=O)NC(c2nn[nH]n2)CC)C)CCCCO1 c1(-n2ncc(C(=O)NCC(C)NC(C(C)C)=O)n2)ccc(Br)cc1 C1(CC)CCC(N(C(=O)CCC(C)NC(c2cccc(O)c2)=O)C)CC1 c1(C(=O)Nc2c(C)nn(C)c2)cnc2ccc(-c3cncc(F)c3)cn12 Cc1cccc(F)c1CC(N1CCCC(NC(=O)CCCCN2CCCC2)C1)=O c1(OC)cc2ccc(N(C)NCCCSc3nccn3C)nc2cc1OC CN1CC2(CCN(CC34CCC(C3)C4(C)C)C2)OCC1=O Cc1cccc(C)c1CNC(=O)CSc1nccn1-c1ncc(Br)cn1 Cc1cc(CCNC(CC(=O)OCC(C)C)=O)c(C)n1-c1ccccc1 C1(N(C(CN(S(CC)(=O)=O)C)=O)C)CCN(C(=O)COC2CCCOC2)C1 Cc1c(C(N2CC(C(N)=O)(CNC(=O)CCC3CC3(C)C)C2)=O)ccn1CCO C12(C(=O)NCC3COCCN(C(CCC=C=C)=O)C3)CCCCCC1OCC2 C1(NC(C2(C(C)NC(C3CC(C)(F)C3)=O)CC2)=O)CCC(N(C)C)CC1 c1(C(=O)NCCN(CC(C)O)C(c2ccccc2)=O)c[nH]nc1C1CCOC1 CC1CN(C(c2ccn(CC(F)F)c(=O)c2)=O)CCCN1C(=O)C(O)CC(N)=O n1(CCC(N2C(CCNC(C3C(=C)C3)=O)CSCC2)=O)ccc2cc(Cl)ccc12 Cc1cccc(OCCCC(=O)N2CCC2CNC(c2ccc(CO)o2)=O)c1 N1(C(C(CO)N(C)C)=O)CCC(NC(C2(C(F)F)CC2)=O)C(C)(C)C1 c1(C(=O)NC2C(CNC(CCC(=O)NC)=O)CCCC2)n[nH]c2c1CC(C)CC2 N1(C(=O)NC(C2CC3(CC3)CO2)CCC)Cc2ccc([N+](=O)[O-])cc2C1 C12(CNC(c3cnc(=N)[nH]c3)=O)CCC(CNC(C3CCCOC3)=O)(CC1)CO2 C(=O)(CS(=O)(=O)NC1CC1)NC(CNC(c1ccn(CCC)n1)=O)CO CCC(CN(C)C)CC(=O)N1CCC(CCNC(c2cnsn2)=O)C1 C1(C2N(C(CCc3c(C)ncs3)=O)CCC2)CCN(C(C2CC23CCC3)=O)CC1 Nc1cc2[nH]cnc2cc1C(=O)NCC(CO)NC(=O)C1=CC2C=CC(C1)C2 c1(CC(N2CC3C(NC(c4c(CC)scc4)=O)C3C2)=O)ccc2c(c1)CCOC2 C1(C(=O)NCCc2cncc(C)n2)(CC)CCCN1C(C1CC=C(C)CC1)=O C(=O)(CC(C(F)F)C(C)(C)C)NCC1N(C(C23CC(F)(C2)C3)=O)CCC(C)C1 c1(CC)ncc(Cl)cn1.n1(CC(=O)NC(CC)CSC)cc(C(C)O)nn1 C#Cc1ccc(C(N2CC(C(=O)OC)C(C(C)C)C2)C(=O)NCC)cc1OC N1(C(CC=C=C)=O)CCCC1(C)CNC(=O)C(C)Cc1ccccn1 C=CCCCCC(=O)N1CC(NC(c2ccc(NS(C)(=O)=O)nc2)=O)CC1CO Cc1cc(Cl)ncc1CC(=O)NC(CNC(=O)C(c1ccc(F)c(C)c1)=O)CO CON1CCC(N(C)C(C2CCN(C(c3ccc(=N)[nH]c3)=O)CC2C)=O)CC1 N1(C(CCSC)=O)CCC2(NC(C34CC(C(C)(F)F)(C3)C4)=O)CC2C1 c1(OCC)ccc(NC(C2CCCN(C(=O)NCc3ocnc3C)C2)=O)cc1 C1(C)(NC(C(C)OCC)=O)CCCN(C(=O)CCC(=O)c2cccc(N)c2)C1 C1(C(=O)OCC)CCOCCN1C(c1csc(-c2ccc(C)cn2)n1)=O Cc1nc(CNC(C2(C)COC2)=O)oc1C(=O)NCC=C1CCSCC1 C1(COC(C2CSCN2C(C2CCC2)=O)=O)(CO)CC1(F)F C(=O)(C1Cc2ccc(F)cc21)NCC1CN(c2nc(C)c([N+](=O)[O-])cn2)C(C)C1 C(=O)(C1=CCCC(C)(C)C1)NC1(CNC(c2nc(CC(C)C)sc2)=O)CCC1 O=C(CCC1=CCc2ccccc21)NC1CCC2(CC1)CN(C(C1COC1)=O)C2 c1(C(=O)NCCC(=C)CNC(c2cnc3nccn3c2)=O)cc(F)c(F)cc1N C1(CNC(C2C(CC)OCC2)=O)CCCCN1C(C1CC2(CSC2)C1)=O C1(NC(C(C(C)O)NC(C)=O)=O)CCCN(C(=O)C=Cc2cncc(F)c2)CC1 N1(C(C(=Cc2ccco2)C)=O)CC2(C1)CN(C(=O)C1=CC3CCCC13)CCO2 Cc1ccc(F)cc1C(=O)N(C(C)(C(=O)NC1CCCC(O)CC1)C1CC1)C C(CN=C(NCC(F)(F)Cl)NC1CCN(c2nc(C)cs2)CC1)SC C=CC1CCN(c2nnc(C3CC3)n2CC2CCN(C(N)=O)C2)CC1 Cc1cc(Cl)cc(C(=O)NC(C)CCNC(=O)Cc2n[nH]cc2Br)c1N C1(NC(=O)Nc2c(C)nn(CC(F)(F)F)c2)CCn2c(Br)cnc2C1 c1(CN(CCC)CCNC(=O)CSC(C)CC)ccccc1CC CCCCCCC(O)CCC(=O)NC1CCCC12CCN(C(C)=O)C2 C1(NC(C=C(COC)C)=O)CCCCN(C(=O)C(C)Oc2ccc(Cl)cc2Cl)C1 C(C(C)(C)C#CC(=O)N(C1CC2CC2C1)C)NC(COC(CC)CC)=O C1(NC(CCCC)=O)(CO)CCN(C(=O)CCC2CCC(=O)NC2)C1 CC(Cc1ccccc1)(CC(=O)O)c1ccccc1.c12ccc(c(F)c1)NC(=O)C2 c1(OC(C(=O)NCC(CNC(c2ccc(OC)o2)=O)C)C)ccc(C)cc1C Cc1nsc(C(N2C(CC(=O)NCCCC(=O)NC3CC3)C3CCCC23)=O)c1N N1(C(=O)C2CCc3snnc32)CCC2(CC1)CC(NC(C1(CO)CCC1)=O)CO2 c1(C(=O)NC2C(NC(=O)C=CC=C(Cl)Cl)C2)cccc(-c2ccccc2)n1 CC(CS(C)(=O)=O)C(=O)NC1(C)CCN(C(c2[nH]nc3ncccc23)=O)C1 c1(C(c2nnnn2-c2ccccc2Cl)NCCOC)cnn(C(C)C)c1C c1(C(N(C2CCCN(C(=O)C(C3CCOCC3)O)C2)C)=O)sc(Cl)cc1Cl C1(C)(C(N2C(COC)CC(O)C2)=O)CN(C(=O)CC2COC(=O)C2)CC1C N1(C(c2c(I)cc(C)c(C)c2)=O)CC2CCN(C(c3[nH]cnc3C)=O)CC2C1 N1(C(C(C)(C2CC2)OC)=O)CCN(C(C2(n3cncn3)CC2)=O)CC12CCC2 c1(C(N(CCCC(=O)NC(C2CCOC2)CC)C)=O)ccnc2cc[nH]c12 C(CC(=O)OC)N(CC(=CC(=O)OC)C)CC=C1CCCC1 N1(C(c2ccc(SC)o2)=O)CCOC2(CCC(NC(=O)C3=CCOCC3)CC2)C1 c1(N2CCC(C(C)NC(COC(CC)C)=O)C2)cc(CCSC)nc(Cl)n1 C1(CNCC(O)COCc2ccc3c(c2)OCO3)CCCC(F)(F)CC1 Cc1cc(CC(=O)N(C2CCN(C(=O)C=CC3(C)COC3)C2)CC2CC2)n[nH]1 C1(C(=O)NC(C2CCN(C(=O)CCc3ccon3)C2)(C)C)OC(C)(C)OC1(C)C c1(C(=O)NC2CN(C(c3n(CC)ncc3)=O)CC2C)c(F)cc(F)cc1Cl c1(C(=O)NCC(CC(C)C)NC(CCc2cc(C)no2)=O)c(Cl)nn(C)c1Cl C1(CNC(=O)CCSc2ccccn2)CCC(NC(=O)C(=O)NCC2CC2)CC1 N1(C(Cc2nc(=N)[nH][nH]2)=O)CC2(CCC(CNC(c3scnc3C(F)F)=O)O2)C1 C1(C)(CNC(COC(CC)C)=O)CN(C(c2cccn3ccnc23)=O)C(C)(C)C1 c1(OC)cccnc1N(C)C(c1cc(C(C)(C)C)c[nH]1)=O c1(C(=O)NC2C(CNC(C(C)(C)S(C)(=O)=O)=O)CCC2)cc2ccnc(Cl)c2[nH]1 C(=O)(C1CCCc2ccnn21)NC12CN(C(CCC)=O)C(CC1)CC2 CC(=O)CC(C)(C)C(=O)NC(C)C=CC(=O)NCC1CC(O)C1(C)C C(=O)(C1=CC2CCCCCC12)N(CCN(C(c1c(CC)cco1)=O)C)C(C)C c1(C(N(CCC(C(C)C)NC(CCCOCC=C)=O)C)=O)cnc2[nH]ccc2n1 c1(C(C(=O)NCC2CCCO2)N(CCNC(C)=O)C)noc2c(Cl)cccc12 C1(CCNC(c2ccc(CCF)cc2)=O)CCCN(C(=O)C(O)C2CC2)C1 Cc1ccc(F)c(CN2CCCC23CN(C(c2cc(Cl)ccc2Br)=O)C3)c1F Cc1cc(NC(C2CC3CC3N2C(c2cc(C(C)C)no2)=O)=O)cc(F)c1Br c1(C(N2CCC(OCCNC(CC(=O)NCC)=O)C2)=O)c2c(c[nH]c1=N)CCCC2 C(=O)(C1=CCCCC1)N1CCC(NC(CN(C(CCCCC)=O)CC)=O)C1 N1(C(C2CCC2)=O)CC(O)C(C(=O)N(C2CC2)CC2CCC2)C1.C1CC1 C(=O)(C1=NOC2(CCOC2)C1)N(CCNC(c1c(C)cc[nH]1)=O)C(C)C c1(C(=O)NC2CC(NC(c3ccc(C4CCC4)cc3)=O)C2)n[nH]c2cccnc12 C1(CNc2cn(CC(=O)O)nn2)CC12CC2(F)F c1(C(=O)NC(C2CCOC2)CNC(c2c(COC)cco2)=O)cnc(Cl)n1C c1(NC(C)CC(C)NC(=O)C(C)(C)CO)ncc(C#N)cc1F C(=O)(CC1OCCc2ccsc21)NCCCC(c1ccccc1)NC(CSC)=O CC(C)(O)C(F)C(=O)NCC(C)(C)NC(c1cn(C2CCC2)nn1)=O N1(C(c2c(CC)ncnc2)=O)CC2CC(NC(=O)CCSc3ccccc3)C1C2 Cn1nnc2c1CC(C(=O)NC1CCN(C(=O)Cc3csc(S)n3)C1(C)C)CC2 c1(C(N2CCCC(NC(c3ccc(Cl)cn3)=O)C2)=O)cnc2[nH]ncc2c1 C(C1c2ccccc2CCN1C(c1cc(COC)no1)=O)NC(C(CC)C#N)=O C(C1CCCO1)=CC(N1C(CNC(C2CCCCS2)=O)CC1)=O C(=O)(C(C(C)C)n1cccc1)N(CCN(C(CC(=C)C)=O)CCOCCO)N(C)C.C Cn1ncc(C(=O)NC2(C(=O)NCC(C)(O)C3CCCC3)CC(O)C2)c1Cl CC(C)C(F)(CNC(=O)C=CCN1CCC1)C(=O)NCC1CN2CCC1C2 c1(C(=O)NCC2CN(C(Cc3cc(C)ns3)=O)C(C)(C)C2)cn2cccnc2n1 c1(C(N2CCC(NC(CCN(CC)CC)=O)C2(C)C)=O)nn(C)c2c1CCCC2 c1(CN(CCNC(c2cnc(C3CC3)s2)=O)CC)nc(C)c(C)o1 C(=O)(C(C)(C)CC(F)F)N1CC2C(CNC(C(CC)C#N)=O)C2C1 C1(NC(=O)C(c2cnccn2)C)COCC1S.C1(C(C)(C)C)CCC1NC(C1CCCC1)=O N1(C(c2c(C)nc(C(C)C)s2)=O)CC(CNC(=O)C=Cc2cnc[nH]2)C(C)(C)C1 c1(COC)cccc(CC(=O)NCC(C2CCC2)NC(=O)C(C)(C)CF)c1OC C(=O)(CCCC(C)C)N(C1CCNC1)C(CSC)=O.c12ccc(cc1)o2 c1(OC)nc(Cl)c(C(=O)NC2CC(CNC(C3(Cl)CC3)=O)C2(C)C)s1 CC1=C(CNC(=O)C(C2(C)CC2)NC(c2c[nH]c(=N)o2)=O)CCC1 C(C(C(=O)NC(C)(CNC(=O)Cc1cnns1)CO)c1ccccc1)SC C12(n3cc(CC(=O)OC)nn3)CCC(C(N3CCOC(C(C)C)C3)=O)(CC1)C2 c1(N(C)CCNC(=O)CC2C=CCC2)ccsc1.C1CCO1 C(=O)(C(C)(C)CC(C)(C)C)N1CCC(NC(C=C(C)Cl)=O)CC1C1CC1 C=CCC(CC=C)C(=O)N1CCCC(CC(=O)NC(CCCC)C(=O)NC)CC1 CS(=O)(=O)CCC(=O)NC(CO)C(N1CC2CSCC2C1)=O C(=O)(C(C)C(F)(F)F)NCC(C)CNC(c1c[nH]nc1-c1ccccc1)=O N1(C(C(c2ccn(C)c2)C)=O)CCCC(C)(C(=O)NCCN2CC3CC3C2)C1 CCC(CC(F)F)C(=O)N1CC2(CC2)CC1CNC(c1cnc2c(c1)CCC2)=O C(C(C(=O)NCCC1CC=CC1)NC(C1CC=CCO1)=O)SCC c1(N2C(CN(C(=O)C(O)CC(C)(C)C)C)CCC2)nc2ncc(Cl)cc2o1 N#CC(CC1CC1)C(=O)NCCN(C1CCCC1)C(c1ccnnc1O)=O CC12CC(C(=O)NC(CNC(C3CCCOC3)=O)C3CC3)(CCO1)C2 C=CCC(C)(C)CC(=O)NCC1(C(N)=O)CN(C(=O)CC2CCOC2)C1 c1(CCC(=O)NCC2C(NC(C(CSC)O)=O)C2)ccnc(C)n1 C(CCCCC(=O)N1CCCCC(CNC(=O)CO)C1)SC c1(C(=O)NCC2C3N(C(C45CC(C)C4C5)=O)C(CC3)C2)cccc2nncn12 c1(C(C)C)cccc(C(N2CC(O)(CNC(=O)C=Cc3cocn3)C2)=O)n1 C(=O)(C(C(C)C)C1CCCCC1)OC(CC)C(=O)N1CCCC1 C1(COC)CN(C(=O)CCn2cnc([N+](=O)[O-])c2)CCN1C(=O)C1=CCCCO1 Cc1nc(CC2CC2)sc1C(N1CC(C(C)NC(c2cnc(S)n2C)=O)C1)=O C=CCN=C(NCc1csc(C(C)SC)n1)N(C)CCOc1ccccc1C C1(OC)CC(CNC(=O)CN2CCS(=O)CC2)N(C(=O)CCc2ncco2)C1 C(=O)(CC(O)C(C)C)NCC(CC(C)C)NC(=O)CC1CCC2(CC1)CC2 C1(C2CCN(C(=O)NC)C2)NC(=O)NC1=O.C1(=O)CN1 C1(C)(C(N2C(CN(C(CC3C(C)OCC3)=O)C)CCC2)=O)CC2(CCC2)C1 C(C)(C(=O)NCC(C)N(C(=O)CN1CCC(=O)NC1=O)C)(C(C)C)NC(C)=O Cc1cc(CNC(C2(C)CCCN(C(=O)CCC3CCCCO3)C2)=O)nnc1C c1(C(=O)NC2(CC=C)CCN(c3ncc(C#N)cc3Br)C2)cn(C)c(C)cc1=O c1(C(N(CCCC#C)CC2CCCC2)=O)ccc([N+](=O)[O-])c(C)n1 CC1C(NC(=O)Cc2csc(-c3ccoc3)n2)CCN1C(C1CCCOC1)=O c1(-c2cncc(C(=O)NCC(=O)NC3CC3)n2)ccc2ccnc(O)c2c1 C12(C(N(C3CCCC3)CCCNC(CN(CCC)C)=O)=O)C(=O)C3CC1C2C3 N1(C(Cn2c(C)ncc2)=O)CCC(CNC(=O)C(O)C2CCC2)C1(C)C N1(C(C2CC(C)N2C(C2(CC=C)CCCC2O)=O)=O)CCC(CF)CC1 CCCCCC(O)CC(=O)NCC(C)(C)NC(=O)Cc1ccccc1C(F)(F)F N1(C(c2cnn(C(C)C)n2)=O)CC2CCC(CNC(c3ccnc(S)c3)=O)C2C1 C(=O)(CS(=O)(=O)NC)N(CCCNC(=O)CC1COCCO1)CC c1(SC)cccc(C(=O)NCC(C)CNC(c2cccnc2O)=O)c1Cl O=C1CC(CC(N2CCC(NC(=O)CCc3cnco3)C(F)C2)=O)CCCN1 C1(NC(C(CCC)OC)=O)(CNC(C2CCC2(C)C)=O)CCC(F)(F)CC1 Cc1cc(C=CC(N2C3CCC2(CNC(=O)C=C2CCC2)CC3)=O)ccc1F c1(C(N2C(CNC(CCc3cncc(C)c3)=O)CC2)=O)ccc2nncn2c1 c1(C(=O)Nc2ncc(-c3ccncc3F)cc2C(F)(F)F)c(Cl)cc(Cl)cc1Br C(C(CC(F)(F)F)NC(=O)CNS(=O)(=O)CCCC)N(C(CCC=C)=O)CC c1(NCC(C(C)(C)C)(F)F)nccc(=NCCCCCc2ccc(F)cc2)[nH]1 c1(C(n2c(CC)ncc2)C)nc(-c2ccc(COC)cc2)nn1CCF C1(NC(=O)CS)CCCC(CNC(c2c[nH]nn2)=O)C1.c1(C2CC2)ccccc1 c1(NCC)cncc(C(=O)NCC2(CCNC(C3CC3C(C)C)=O)CC2)c1 N1(C(CC(CCCC)NC(=O)CC=C(Cl)Cl)=O)CCCN2CCCC2C1 Cc1nc(CCCC(=O)N(C)CC2CCCN2C(=O)C(C)c2ccsn2)cs1 C#CC1CN(C(=O)C(n2ccc(C)n2)C)CCN1C(=O)C(C=C)OC C(=O)(C(C1=CCCCCCC1)N(CCCO)C(C)C)NCCCC N1(C(C(C=C)C)=O)CCN(C(=O)CCC(C)OC)C(c2ncc[nH]2)C1 C1(C)(NC(C(C)OC)=O)CCCN(C(=O)CCc2ccc(C)s2)C1 c1(C(N2CC3(CCN(C(CC(CCC)C)=O)C3)C2)=O)cnc2c(c1)CNC2=O c1(C(=O)NCC(O)CNC(C2(F)C3CCCC23)=O)ccc2sccc2c1 N1(C(C(C(C)C)NC(N)=O)=O)CCOC2(CCN(C(c3ccccc3)=O)CC2)C1 CC1(NC(=O)CCc2csnn2)CCCN(C(C2CC(=O)OC2(C)C)=O)C1 C1(OC)CC(CCNC(=O)CNC(=O)Cn2ncnn2)C1 c1(C(N2CCC(CNC(=O)Cc3cccnc3)C23CC3)=O)cnc2cc[nH]c2c1 c1(NC(C2CCCN(C(C(C)C3CC3)=O)CC2)=O)ccc2c(c1)CCO2 c1(SC)nc(O)nc(C)c1C(=O)NC1CCCC1NC(=O)CC(C)n1cccc1 C(C1C(=O)N(C2CN(C(=O)C3=CCC3)C2)CC(=O)O1)OC(C)=O.C(C)(C)(C)OC c1(C(N2CC(C)C(O)CC2)=O)noc2c1CN(S(=O)(=O)C(C)C)CC2 c1(CN2CCC(C(N3C4CCC3COC4)=O)C(O)C2)c(F)cc(Cl)cc1Cl N1(C(C2(F)C(C)C2)=O)CCC(CO)(NC(=O)CCCc2nccs2)C1 Cc1cc(C(=O)NC2C=CC(CC(=O)NCc3ncnn3C(C)C)C2)cc(O)c1 N1(C(C2CC3C=CC2O3)=O)CC2(CCC2)C1C1CCCO1 N1(C(CNC(=O)OCC)=O)CCC(C(=O)Nc2cn[nH]c2)C(C)(C)C1 Cc1cccc2c(C(N3CC(NC(=O)C(F)(F)C(C)O)C4CC34)=O)c[nH]c12 CC1(C)CC(C)(CNC(=O)C(F)CC2CCC2)CN1C(c1c[nH]cc(Cl)c1=O)=O Cc1nn(C)nc1C(=O)NCCOC1CCN(C(=O)C(c2c(C)n[nH]c2C)C)C1 c1(C(N2CC(C)(C(N(C)CC3(O)CCCCC3)=O)C2)=O)ncncc1Cl C(=O)(C1=CC(C)(C)C1)N(C(CNC(c1ccnn1C)=O)C1CC1)C c1(C(N(C2CCN(C(C3CCC3(F)F)=O)CC2)CCC)=O)cc(C)[nH]c1C CN1CCOC(C(=O)NCC23CC(CN2C(c2cc[nH]c(=N)c2N)=O)C3)C1=O C12(CNC(c3ccncc3C(F)(F)F)=O)CC(CN1C(C1(CCF)CC1)=O)C2 C(CC(C(C)(C)C)NC(C1(C)CCCOC1)=O)N(C(CNC(CC(C)C)=O)=O)C Cc1ccc(C(=O)NC2CCCN(NC(C3CCC(C(N)=O)O3)=O)C2C)c(C)n1 O=C(CCCCCCN(C(=O)COc1ccccc1)C1CC1)NC1CCC1 N1(C(c2cc(C)c(Cl)cc2)=O)CC2(C1)CN(C(=O)C(C)O)CC(C)(C)O2 c1(C(=O)NC23CCCC2N(C(=O)Cc2cccs2)CC3)cc2cncn2c(O)n1 C1(CNC(C=CC(C)(C)SC)=O)CN(C(=O)CC2CCN(C)CC2)CC12CC2 C1(C(=O)NCc2c(C(N(CC#C)C3CC3)=O)cco2)C2CCC(F)C12 c1(C(N2CCC(C(N3CCCC(CC=C)C3)=O)(OC)C2)=O)ccc(C#N)c(C)c1 CC1C(NC(c2nnc(O)nc2O)=O)CCCN1c1ncnc(Cl)c1F Cc1cc(C)c(C(=O)NC(CC2CC2)C(=O)NCCOCC2CCCC2)cn1 N1(C(c2c(SC)ccs2)=O)CCC(NC(=O)CC2CCCN(C(C)C)C2)CC1C C1(C(=O)NC(C)C(C)NC(c2cn(CCC3CC3)nn2)=O)CC(F)C(=O)N1 O=C1CN(CCCOCC(F)(F)F)C(=O)N1CCC1CC=CCC1 C1(CC)(CC)CC(NC(c2cc3scnc3[nH]2)=O)CN1C(=O)Cc1nocc1C c1(C(N(CC(O)CNC(c2c(Cl)cnn2C)=O)C)=O)coc2c1CCCC2 N1(C(C=C(C)C)=O)CCCC(C)C1CCNC(C12CC(F)(C1)C2)=O C(CC(C(C)(C)C)NC(=O)CC1(C)CC1)N(C)C(C1CC(=O)OC1(C)C)=O N1(C(c2cn(C)c(=O)n2C)=O)CCCCCC(NC(C2CC23CCSCC3)=O)C1 CC1(C(=O)NCC2CCC(O)CC2)CCN(C(=O)Cn2[nH]cnc2=N)C1 C1(NC(COCCC)=O)CN(C(=O)CC2CC2C2CC2)C2CCCC12 C(=O)(C(F)(F)C(F)F)NC1C(C(=O)NCCc2nccs2)COCC1 CC(C)C(CCN(C)C(C1CC(C)(C)C1C(F)(F)F)=O)NC(c1cnco1)=O N1(C(C(C2CCCCC2)C)=O)CCC(NC(c2cnccn2)=O)C1C c1(C(=O)NCC(F)CO)ccn(C)c(=O)c1.C1CC(=O)N1CC c1(C(C)=O)ccccc1C(=O)NC(CNC(=O)C(F)Cc1ccccc1)C1CC1 C(c1ccccc1F)=CC(=O)NC1(CNC(c2cc(C)c(C)o2)=O)CCC1 C=C(Br)CC(=O)NC(CN(C(=O)CN(C(C)=O)Cc1ccco1)C)CC c1(C(=O)NC2CC(CCNC(CC(C)(C)O)=O)C2)cccc([N+](=O)[O-])c1Cl Nc1csnc1C(=O)NCC1CCCC1NC(c1csc(-c2cccnc2)n1)=O c1(C(=O)NCCN(C)C(C2CCCC3(CCC3)C2)=O)cc2scc(Cl)c2[nH]1 C(=O)(CS(=O)(=O)NC1CC1)NCC(C)NC(C1(N(C)C)CC1)=O C(C(C(=O)NCc1ncc(C)cc1C)C(C)(C)C)NC(C(C(CC)C)=O)=O Cc1nn2cccnc2c1C(N1CCN(C(=O)CCC2CC2)C(C2CC2)C1)=O C(CCCCC(=O)NC1C2CN(C(C3(C)CCCOC3)=O)CC12)OC N1(C(=O)OC(C)(C)C)CCC2C(C1)CN2C(=O)CCNS(C)(=O)=O CC1CN(C(C2(N3CCCC3)CCC2)=O)CC(C)CN1C(=O)C1=CCCCO1 C=CC1(C(N2CCOC(C(N)=O)C2)=O)CCN(C(c2cc(CC)oc2C)=O)C1 C(=O)(C(CC(C)C)N1CCCC1=O)NC1C(c2cn(CCC=C=C)nn2)CCCC1 C1(NC(Cc2c(C)con2)=O)CN(C(=O)CN(C)S(N)(=O)=O)CC1C N1(C(CCOC)=O)CCC2CC12C(=O)NCCC1CC1C1CC1 Cn1ncc(Br)c1CN1CCCC(NC(C2(C)C=CCC2)=O)C1 C(=O)(C(C)CCNC(=O)CC(COC)NC(C1CCO1)=O)OC CC(C(F)C(=O)NCC1CN(C)CCN1C(=O)Cc1csnn1)C(F)(F)F N1(C(C(C(C)(C)C)OC)=O)CC2CCN(C(=O)CCn3cnnn3)CCC2C1 N1(C(c2c(C)n(C)cc2)=O)CCC(CNC(=O)C(C)CN2CCOCC2)C1(C)C C(=O)(C(C)C1=CCCC1)N1CC(CC)N(C(c2nccn2CC)=O)CC1 Cc1c(C(N2CCC(CN(C(=O)CC(C)CF)C)C2)=O)csc1Br C(=O)(CCCCCC(C)C)NC1CCN(C(CCCCC(=O)NC)=O)CC1(C)C c1(C(N2C(CNC(C=C(C)C)=O)C=CC2)=O)ccc(N2CCC(C)(C)C2)cc1 C(C(F)(F)C(=O)N1CCN(C(C2(F)CCN(C(C)(C)C)C2)=O)CC1)OC CC(C)C(F)(F)CCNC(=O)CC(c1ccccc1)C1CC1 N1(C(CCC#C)=O)CCCN(C(c2ccc(CC)[nH]2)=O)C(C)C1 CCC1=C(C(=O)N2CC(C3CCN(C(c4ccc(C)c(C)c4)=O)C3)C2)CCCO1 O=C(C1=CCCCO1)NCCC1(NC(=O)COc2cncc(Br)c2)CCC1 N(C1CCc2cccnc21)C(CC1OCCN(C(C(CC)N(CC)CC)=O)C1)=O C=CCCCCCCC(=O)N1CC(F)CC1C(=O)NCC1CCC(CO)O1 c1(C(N2CCOCC2C(C)C)C(=O)NCC)ccc(C(C)C)cc1F C1(C(N(C2CN(C(C3CCN(c4nccn4C)C3)=O)C2)C)=O)CCC(C)(C)CC1 C(=O)(C(F)C(C)C)NCC1(NC(C2CCC(=O)NC2)=O)CC(OC)C1 N1(C(c2c(C)nn(CCO)c2)=O)CCN(C(=O)C(C)(O)C2CC2)C2(CC2)C1 C(=O)(C(CNC(C1CCC1C(N)=O)=O)N(C)C)NCC(=O)NCCC C1(CNC(C2(C)CCC(C)C2)=O)CN(C(=O)CC2CCC(C)(C)CO2)CCCO1 C1(CC)(CC)NC(=O)N(CC(=O)N(C)CCNC(C2CC23CC(F)(F)C3)=O)C1=O C1(N(C(=O)C(N)=O)C)CS(=O)(=O)C12CCN(C(C1CC(CC3CC3)C1)=O)CC2 C1(C(=O)OC)CCC(C(=O)N(CC(C)(C)CNC(C2CCCN2C)=O)C)CC1 C=CC1(C(N2CC(C)(C(=O)OC)C2)=O)CCN(C(=O)CC2C=NN(C)C2=O)C1 C(CC(F)F)(C(=O)NC1CCS(=O)CC1)N(C(C1CC(C)(CC)C1)=O)C C=CCC(F)(F)C(=O)NC(C)CCNC(c1cnn(-c2ccc(OC)cc2)c1)=O c1(CN2C(C(N3CCOC(C(F)(F)F)C3)=O)C(O)CC2)cc(O)c(O)cc1O CC(C)(C)C1=NOC(CNC(=O)NCCSCc2ccco2)C1 n1(CCCC)ccc(C(=O)NC(CNC(=O)Cn2ccnc2C(C)C)CO)n1 C=CCCCCCCC(=O)N(C1CCCN(C(c2nnn(C)c2C)=O)CC1)C c1(C(=O)NC2CN(C(CCNS(CC)(=O)=O)=O)CC2C)cc2cnccc2o1 c1(Cc2c(OC)cccc2)cc(=NC2COc3c(Cl)cccc32)cc[nH]1 C12C3CC1N(C3)C(=O)c1ccc(cc1)CC(=O)NC2=O.c1(OC)cn(COC)nn1 Cc1c(C(N2CCCN(C(C34CC(C(F)(F)F)(CO3)C4)=O)CC2)=O)cccc1O C1(C(=O)NCc2c(CC)nns2)CCC2(CC2)N1C(C1COCC(C)O1)=O N1(C(C2(NC(c3c[nH]c(=NC)s3)=O)CCCC2C)=O)CCN2CC(C)CC2C1 CCC(C)C(O)C(=O)N1CCCCC(NC(c2ccnc(Cl)c2N)=O)C1 O=C(N=c1cc2ccccn2[nH]1)C1CC(O)CN1Cc1ccc[nH]1 n1(CCC(=O)NCC(CN(C(=O)CCS(C)=O)C)O)cnc2c(cnn2C)c1=O C=C(C)CC(C)C(=O)NCC(C1CCN(C(C2(n3cc(Cl)cn3)CC2)=O)CC1)C Cc1ccc(C)c(C(=O)C(C)OC(c2cc(C)no2)=O)c1 CCCCC(C)CCC(=O)N1CCC(C)(NC(=O)Cn2nnnc2C(C)C)C1 Cc1nn(C)cc1C(=O)N(C1CCC(n2cc(-c3ccccc3I)nn2)CC1)C C1(OC)CN(C(c2oncc2C)=O)CC1NC(=O)CC1CCC(C(C)(C)C)CC1 C1(NC(C2N(CC)CC2)=O)CCN(C(=O)CCC(C)C)CCC1CO c1(C(N2CCN(C(c3n(CC)ccn3)=O)C(C(F)F)C2)=O)cnc2sc(C)cn12 c1(C(N(C)CC2(NC(C3CCCC3)=O)CC2)=O)csc(-c2cccs2)n1 CC1CC2(CCN(C(c3cc(O)cc(F)c3F)=O)CC2)CN1C(C1CC1(Cl)Cl)=O O=C(CN1C(=O)Cc2cc(F)ccc21)NCC1CCN(C(c2cscn2)=O)C1 Cc1c(C(=O)NCc2csc(C(=O)NCc3nccc(O)n3)c2)[nH]ccc1=O N1(C(C(C)CN2CCOCC2)=O)CCCN(C(=O)CCCC(F)(F)F)C(CO)C1 C(CCCCC(=O)NC(C)C(C)NC(c1cncc(C)n1)=O)NC(C)=O c12ccc(cc1)s2.c1(C(N2CCC(C3CCCN3C(=O)C3CC3)C2)=O)csc(S)n1 N1(C(C(CC(C)C)=O)=O)CCC(C(=O)NCC2(CCCO)CC2)C12CCC2 Cn1cc(CN2CCCC2C(=O)N(C)C)c2ccc(F)cc12.C12(CCC1)CC(=O)N2 CCC(C)(CC)C(=O)NC1CCC1NC(=O)CCc1ccc(C(=O)OC)cc1 N1(C(Cn2c(C)nnn2)=O)CC2(CCC(CNC(C3(CO)CCCO3)=O)O2)C1 c1(C(C)NC(=O)NCC(C)Cn2ccnn2)cc(F)cc2c1OCOC2 C(CC(C(=O)NCCC(C)SCC)NC(c1nnccc1C)=O)=CC N(S(=O)(=O)N1CCNC(C)C1)(C(CC)CC)CCC(C)C c1(CCC(=O)NC2CN(C(C3COCCO3)=O)CC23CC3)cc(F)cc(F)c1 C(=O)(CC(O)C(C)CC)NC1CCC(CCC(=O)NCC=C)C1 c1(CCNC(C2(C)COCC2(F)F)=O)c(Br)c(O)c(O)c(Br)c1Br C1(CNC(C2(SCC)CC2)=O)C(C2CC2)CCN1C(c1ncc(C(F)F)s1)=O N(C1CCCc2c(F)cc(Cl)cc21)C(C1NCC(=O)NC1)=O c1(C(=O)NC(C2CCCN(C(C3(C(F)F)CCCC3)=O)C2)C)cc(C#N)n(C)n1 c1(C(=O)NC2CN(C(c3c(CC)nns3)=O)CC2C)ccc(Cl)nc1OC C1(C(=O)NC(C(C)C)CNC(c2ccc(Cl)o2)=O)CC2CCC1CC2 c1(C(=O)NC(CN(C(=O)Cn2nccc2C)CC)C)ccc(P(C)(C)=O)nc1 C1(O)(CNC(COc2cc(C)on2)=O)CCN(C(C2(O)CC2)=O)C1 c1(C(=O)OC)ccnc(C(=O)NCCC2(CNC(C3COC(C)(C)C3)=O)CC2)c1 C1(CCC)(NC(c2ccc(OC)cc2F)=O)CCCN(C(c2coc(C)c2)=O)C1 c1(C(=O)NCC2CN(C(c3cncc(OCC)c3)=O)C2)cc(F)c(OC)c(Br)c1 c1(NCCCC=CC)ccc(S(=O)(=O)N2CCCC(C(C)(C)C)C2)cc1Br c1(CCNCC2CC(C(C)(C)C)C2)ccc(F)cc1Br CCC(C)C(CNC(=O)CN(C(c1ccc[n+]([O-])c1)=O)C1CC1)CO Oc1nc(CNCC(N2CCCCC2)c2cccs2)cc2ccccc12 C1(C(=O)NC(C)C(C)(C)NC(c2cccc(-n3cnnn3)c2)=O)COCCOC1 C1(CNC(C=CC(CC)C)=O)COCCN(C(c2cc(CC(C)C)[nH]n2)=O)C1 Cc1ccc2occ(CC(=O)NC34CC3CN(C(=O)CN3CC5CC5C3)C4)c2c1 c1(OCC)ccc(CNC(C2CC(O)(CNC(c3cc(OC)n[nH]3)=O)C2)=O)cn1 C1(NC(C2(OC(C)=O)CC2)=O)CCCCN(C(=O)Cc2c(O)ncnc2O)C1 c1(OC)c(F)cc(F)c(N2CC(OCCNC(=O)C(C)C(C)C)C2)c1[N+](=O)[O-] CC1=CCC(C(N2CC=CC(NC(=O)C=CCn3cncn3)C2)=O)CC1 N1(C(c2c(OC)cccc2Cl)=O)CC2COCCC2(NC(c2ccco2)=O)C1 C(CCCCC(C(=O)NCc1nnn(C)n1)N1CCN2CCCCC2C1)OC C1(CCCC)CN(C(c2nn(C)cc2Cl)=O)CCN1C(=O)C(n1cc(Cl)cn1)C N1(C(C(C2CC2)OC)=O)CCCC2(CCN(C(c3ccn(C(C)(C)C)n3)=O)C2)C1 CC1CN(C(=O)CCCCNC(=O)CCC(C)(C)C)CC(C)N1C(N)=O CCCCCCCC(=O)N1CCC(NC(c2cc(Br)cnc2N)=O)C1 Cc1ccnn1C=CC(=O)NCCC1CN(C(=O)C=Cc2cn(C)nn2)CCO1 c1(C(CC)=O)ccc(C(=O)NC2(C)CC(NC(=O)CC=C(Cl)Cl)C2)cc1 c1(NC(C=CC2(C)COC2)=O)ccnc(-n2cccc2)c1 c1(C(=O)NCCCCC(C)NC(c2c(Cl)cccc2Cl)=O)cccc(S(C)=O)c1 CC(C)(C(=O)NCCCNC(=O)C1=CC2CC=CCC12)C1=CCSCC1 C1(NC(c2cn(C)nc2)=O)CN(c2ncc3c(ncn3C)n2)Cc2nccn2C1 S(=O)(=O)(c1cccc(C(C)(F)F)c1)N1CCN(c2ccc(OC(C)=O)cc2)CC1 Cc1ccn(C)c1C(=O)NCc1ccoc1C(=O)NCC#CC(F)(F)F N1(c2nc(C(C)C)nc(N3CCC(C#N)C3)c2)CCn2ncc(Br)c2C1 c1(N(CCCNC(C(C=C)O)=O)CC)cc(Cl)ncn1 N1(C(CNC(CCC)=O)=O)CCCC2(CCN(C(C3OCCO3)=O)C2)C1 C1(NC(CCCCCOCC)=O)CN(C(C2CCOC2)=O)C2(CCCC2)C1 N12CCN(CC1)C(=O)C(C)C2=O.C1(CNC(C)=O)CCCOC1c1ncc[nH]1 N1(C(CCN(CC)CC)=O)CC(NC(=O)Cc2sc(O)nc2O)CC12CCOC2 CCCC(C(=O)NC(c1ccccc1)C(=O)NCCc1cncs1)NC(C)=O N1(C(C2C(NC(CCC=C(C)C)=O)C2(C)C)=O)CCC(F)(F)C(O)C1 C(=O)(CC(C)CC(C)(C)C)N1CC(C)(OCC(=O)NC(CC#C)CO)C1 Cc1cc(C(=O)NCC(F)CNC(=O)CC2CC(C(F)F)C2)no1 C1(C(N(CCC(=O)NC2CC2)C)=O)CCN(C(=O)C(C)(C)C)C(C)(C)C1 c1(C(=O)NCC2(CNC(C3(C#N)CC4CC4C3)=O)CC2)onc2ccccc12 N(C(=NCC(C)C)NC1CCCN(C(c2ccccc2)=O)C1)CC1(C#C)CC1 N1(C(C2C(NC(c3cc(O)ccc3Cl)=O)C2)=O)C2CCCC1COC2 C1(C(=O)NCC(CC)NC(c2ccc(SC(F)(F)F)cc2)=O)COC(=O)N1C CC1(C)CC(O)CN1C(=O)C(=O)NCC(N1CC(C(=O)OCc2ccccc2)C1)=O C1(C)(C(=O)NC2(COC)CCC2)CN(C(=O)C(C)Oc2cccnc2)C1 C1(CC(=O)NC2CC(C)(CNC(c3cn(CC=C)nc3)=O)C2)CC(=O)NC(=O)C1 C1(CN(C)C(C2(C)CC2(F)F)=O)CCN(C(=O)CN(C)C2CC2)C1 c1(OC)cnc(C(F)(F)F)cc1NC(c1csc(Cl)c1Br)=O C(=O)(C1=C(C)OCCC1)NC(CCOC)CNC(=O)CC1(O)CCC1 N1(C(c2c(C)n(C)cn2)=O)CC2CC1CN2C(=O)CCC1CCCC(O)C1 c1(C(N2CCCC(NC(c3c(C)noc3)=O)CC2)=O)cccc2c1C(=O)NC2 c1(C(N(CCCC(=O)Nc2ncc(C(N)=O)nc2)C)=O)cccc(O)c1Cl C1(C(=O)NCCCC(C)NC(=O)CN2CC3CC3C2)CCCCN1C c1(C(=O)NCC2(C(F)F)CCN(C(C3C(C)C3)=O)C2)cc2c(Cl)c(Cl)ccc2[nH]1 C1(CNC(c2c(CC)cno2)=O)CCCN(C(=O)Cn2cnc([N+](=O)[O-])c2)CC1 C12(CNC(C3(CNC(C(F)OC)=O)CC3)=O)CC1CN(C(C)=O)C2 C1(NC(CC)=O)CC2CC1CN(C(c1ccnnc1C)=O)C2 c1(C(N2C(CCCNC(c3cnccn3)=O)CCCC2)=O)cnc2n1CCOC2 N1(C(COCC=C)=O)CCCN(C(C2CC(C3CC3)=NO2)=O)CC1C c1(C(N(C2CCN(C(CC3ON=C(C)C3)=O)CC2)C)=O)ccc(=O)n(C)c1 Cc1cccc2[nH]cc(C(N)C(=O)NC3CC3)c12 C1(C(N2CCC(CC(=O)OC)C2)=O)CC12CC(NC(C13CCC(C1)C3)=O)C2 CCCCC(C(=O)NCc1cc(C)c(C(=O)NCCC(C)(C)F)o1)N(C)C C(=O)(CCC#Cc1ccccc1)NC(C1(O)CN(C(C2(O)CCC2)=O)C1)C N1(C(CCc2c(C)ncnc2O)=O)CCC(C2CC2)C1CNC(=O)C1CC1 N1(C(c2ccns2)=O)CC2CCCC(C1)N2C(c1cnon1)=O C1(C(=O)NC(CNC(c2sc(CC)c(C)c2)=O)C(C)C)CC2CC1C1C2C1(F)F c1(C(C)=O)cc(CCC=CC(=O)NC2COCC2NC(=O)C(=O)N(C)C)oc1C c1(C(N(CCCCN(C(C(CC#C)C2CC2)=O)C)C)=O)ccc([N+](=O)[O-])s1 c1(C(N2C(C)CC(NC(=O)CNC(N)=O)C2)=O)ccnc2c(C(N)=O)cnn12 C1(CNC(C2CCCN(CCC)C2)=O)CC(N=c2[nH]n3cc(C)nc3s2)C1 N1(C(C2CCCCC2O)=O)CCC2CN(C(C3CC(O)C3)=O)CC2C1 C1(CNC(C2CCCC(C(F)(F)F)C2)=O)(CO)CCN(C(=O)C(F)F)CC1 C(CC(CC)C(=O)NCC12CC1CN(C(=O)C(F)(F)CO)C2)=CC c1(C(=O)NC(CC)CNC(=O)CC2(O)CCOC2)cnn(CCO)c1C1CC1 S(=O)(=O)(c1ccc(Br)c(F)c1)N1C(C(N=c2c(C)c[nH]cc2)=O)CSCC1 N1(C(CCCOCC=C)=O)CCN(C(c2cnc(C(C)OCC)s2)=O)CC(O)C1 C1(NC(CC(=O)N(C)C)=O)CCN(CCNC(C2CC(C)(C)C2)=O)CC1 c1(C(=O)NCC(N(C)C(C2CC2C(F)F)=O)C2CC2)cccc(Br)c1 C1(C(=O)NCC2CN(C(c3ccsc3Cl)=O)CCO2)C2CCC3C(C2)CC13 Cc1oc(C(C)C)cc1C(N1CCC(O)(CCNC(C2CNC(=O)N2C)=O)C1)=O c1(OC)ccc(C)cc1N1CCC(Nc2nnc(Br)c(C)c2C)C1 CC(C(O)C(F)F)NC(=O)C=CC1CCCN1C(C1CN(C2CCC2)C1)=O CCC(CC)C(C)C(=O)NCC(C(=O)NCCSC)OC c1(C(=O)NC(C2N(C(C(C)OCC)=O)CCC2)(C)C)cccc(OC(F)(F)F)c1 N1(C(c2n(C(C)C)ncn2)=O)CCN(C(=O)C=Cc2ccnn2C)C(C)C1 N1(C(c2c(C)snn2)=O)CC2(C)CC1(C(N1CCCCC(C)C1)=O)C2 c1(C(=O)NCCN(C(=O)CC2CC23CC3)C(C)C)ccc(CN(C)C)o1 CCC(CCCC(=O)N1Cc2ccccc2C1)NC(C1CCCN(CC)C1)=O N1(Cc2cc(-c3c(OCCC)nccc3)n[nH]2)CCN2CC(OC)CC2C1 C1(O)(CNC(CCN(S(C)(=O)=O)C)=O)CCCN(C(=O)C(C)C)CC1.C1C(=O)N1 N1(C(c2c(OC)ccs2)=O)CCC(NC(=O)CC2(OC)CCCC2)C2(CCC2)C1 N1(C(c2cc(C)sn2)=O)CCCCC(C2CN(C(C3C4CCC(=O)C34)=O)C2)C1 c1(CC)ncc(C(=O)NC(C)C(C)NC(c2oncc2C)=O)s1 c1(C(=O)NCC2CCC(NC(c3c(C)ncnc3)=O)C2)ccc(OCF)c(F)c1 C1(NC(c2c(OC)cc(C)s2)=O)C(C)CCN(C(c2csc(C)c2)=O)C1C S(=O)(=O)(c1cccs1)NCCN(C(=O)C(=O)NC1CCN1c1ccccc1)CC C1(F)(C(N2CCC(C(C)(C)C(=O)N3CC4CC4C3)C2)=O)CC=CCC1 N1(C(C2(C)CCCC2)=O)CCOC2(CCN(C(C3CC4CSCC(C3)C4)=O)C2)C1 c1(OCc2nc(-c3scc(C)c3)n(CC(F)(F)F)n2)ccc(C)cc1C c1(C(N2CCC(c3cc(C(=O)OC)on3)CC2)=O)cnn2c1S(=O)(=O)CC2 N1(CCCCCNC(C(C2CCCC2)OCC)=O)CCN(C(=O)C(C)(C)O)CC1 C(=O)(C1CCc2nccn21)NCC1CC(NC(c2nc3ccccc3[nH]2)=O)C1 N1(C(CCC(=O)OCC)=O)CCC(C)(C)C(NC(=O)Cc2c[nH]nc2O)C1 C1(N(CCNC(=O)CCNC(C2CCC2)=O)C(c2c[nH]cc2Br)=O)CCCCC1 C12(C(N(C)CC3C(C)OCC3)=O)CC(CN(C(=O)CCCCC3CC3)C1)C2 CC1(F)CN(C(=O)CC2(C)CC2(Cl)Cl)CCN(c2ncc(Cl)c(O)n2)C1 C1(C(=O)NCCOCCNC(c2c(C)nc(C)o2)=O)COc2ccc(F)cc2C1 n1(CC(C(C)C)(C)O)cnc2c(N3CCCCN(CCO)CC3)ncnc12 c1(NCc2ncc(NC)nc2)nc2ccccc2nc1N1CCC(N2CCC2)C1 Cc1c(C2CCCN2C(=O)NC2(C)CCCOC2)cccc1Br CCC(C)(C)CCCC(=O)N1CCN(CCCNC(C2(C)C=CCC2)=O)CC1 C1(NC(C(C=CCCC)O)=O)CCCC12CN(C(c1ccc(CO)c(Cl)c1)=O)C2 c1(C(N2CCC(C(C)(C)NC(c3cccs3)=O)CC2)=O)ccc(F)c(Cl)c1 N1(C(C2(CC=C)CC=CC2)=O)CCOCC(CNC(=O)CC2COCCO2)C1 N1(C(C2N(C(C)=O)CSC2)=O)CC2CC(NC(=O)C(C)C(C)(C)C)CC1C2 N1(CC(=O)N(CC(O)CNC(=O)CCC2OCCO2)C)CCCCC1=O Cc1cccc2[nH]c(C(=O)NC(C(C)NC(=O)Cc3cnsc3)C(C)C)cc12 N1(C(C=CC(=O)OCCCC)=O)CC2C(CNC(=O)C(c3cncnc3)C)C2C1 c1(C(N2CC(NC(=O)C=CCn3cncn3)C(O)C2)=O)cc(F)cnc1O c1(CC(N2CC(NC(C3N(CCC(C)C)CCC3)=O)C2)=O)nc2ncccn2n1 CC(C)CC(CNC(C1(C#N)CC1C)=O)C(=O)N1CCn2cnnc2C1 c1(NC(=O)NC(CC)C(F)F)cc(C(C)(C)C)ccc1OC c1(C(N2CCCC(NC(c3cccnn3)=O)C2)=O)cc(Br)ccc1OC(F)F c1(CNC(C2C(CNC(C(C)=CC3CC3)=O)CCO2)=O)c(C)n[nH]c1C N1(CC(=O)NC(C)Cn2cncn2)CCN(C(c2cc(F)c[nH]2)=O)CC1 CC12CN(C(c3ccc(CO)cc3)=O)CC1CN(C(C1CC1CF)=O)C2 N1(C(C(c2ccc(Cl)c(Cl)c2)C)=O)CCCC(CO)(NC(c2cnnn2C)=O)C1 C1(CNC(C(C=CC)O)=O)CC2CCC(C1)N2C(=O)C(C1COC(C)(C)O1)O N1(C(c2cnc(=N)[nH]c2)=O)CCC2CN(C(C3CC34CCOCC4)=O)CCC12 c1(C(=O)NC(CC2CN(C(C(C)(C)OC(C)=O)=O)C2)C)cnc(S)nc1 c1(CNC(=O)NCc2scc(C(c3cccc(O)n3)C)c2)nn(C)c(=O)n1C Cc1nc(-c2ccco2)cc(=NCC(C(C)(C)C)NC(C2CC2C)=O)[nH]1 c1(C(=O)CSc2c(F)cc(F)cc2F)ccc2sccc2c1 CCC(CC(F)(F)F)NC(=O)CC1COCCN1C(=O)C(c1cccn1C)=O O=S(=O)(c1ccc(O)c(F)c1)NCS(=O)CC1CC1.C1(OCC(F)F)CCOCC1 C(=O)(CCC(F)(F)F)N1CCC(C(=O)N(C(C)CC2CC2)C)(OC)C1 c1(CC(N2CC(c3nc(C(C)C)[nH]n3)OCC2)=O)ccc(Br)c(C(F)(F)F)c1 Cc1cc(OCC(=O)NCCC2(NC(C3CC3C3CC3)=O)CC2)cc(C)c1 C1(NC(C(CC)NC(N)=O)=O)CN(C(c2ccc3nc[nH]c3c2)=O)CC2(CC2)C1 c1(N(C(C2(O)CC2(n2cnc3cncnc23)C)=O)C)n[nH]c2cc(Cl)ncc12.CC C1(C(=O)NC2CC(NC(c3cc(Cl)cc(C)c3O)=O)C2)CCc2nnc(O)n2C1 c1(CCC(=O)NC(CC)CNC(=O)C(C(=O)OC(C)(C)C)SC)c(C)n[nH]c1C C1(OC)CNC(C)(C(=O)NCC2CCCN2CC(C)C)C1 C12(C(N(CC(C)N(C(CCN(CCCCC)C)=O)C)C)=O)CC(F)(C1)C2 N1(C(C2CCN(C(C)C)CC2)=O)CCN(C(=O)CC(C)(C)C)CC1CCO c1(C(=O)NC2CCCN(C(CS(=O)(=O)NC)=O)C2)c(C)nc2sc(C)cn12 CC1CN(C(=O)C=C(Cl)Cl)C(C)CN1C(=O)CN(C1CCC1)C C1(C(c2nnnn2CC2CCOC2)NCCNC(C)=O)(COC)CCCC1 CC(CC(F)F)C(=O)NC1CCC(CNC(C2CCOC2C2CC2)=O)CC1 CCC(C)CC(C(=O)N1CCCC(F)(F)C1)NC(c1ccc(CF)cc1)=O N1(C(C(CC)(C)C)=O)CCCCC12CN(C(C1CC1(F)F)=O)C2 N1(C(C(N)Cn2cccn2)=O)CCCCC1CCCO C(CN=c1ccc(S(=O)(=O)NC(c2ccccc2)C)c[nH]1)N1CC(CC)OCC1 C1(NC(C2CC23CCN(C(c2ccsn2)=O)C3)=O)COC2(CCCC2)C1 n1(CC(N2C3CN(S(=O)(=O)Cc4ccc(Cl)cc4)CC23)=O)cnc2ccccc12 C(=O)(N(CCC(=O)N1CC2(CCNC2=O)C1)OC)c1c(CC)[nH]cc1 C1(NC(c2c(C)occ2)=O)CN(C(c2cc(C)n(C(C)C)n2)=O)C2CCCCC12 Cc1cc(C(=O)NCC(O)CC(=O)NCC2(C(N)=O)CC2)cc(F)c1 N1(C(CC2(C)CCCC2)=O)CCC2CN(C(c3ncc(Cl)cc3Cl)=O)CCC12 C1(=CC(=O)NC2CC(F)(CNC(c3cccc(N)c3)=O)C2)CCCCCC1(F)F C1(C(=O)NC(C)C(=O)NC2COC(C3CC3)C2)CCCCC1O CCCC(CC)S(=O)(=O)N(C(c1ccc(Br)cc1)C(C)C)C c1(C(N(C(CNC(C(CC)O)=O)C)C)=O)csc(C)c1C C(c1cccc(Br)c1)=CC(=O)NC1(CO)CN(C(C2CN(CC)C(=O)C2)=O)C1 n1(CC(=O)NC(C(C)(C)C)CNC(C2CC2C#N)=O)ccc(=O)c([N+](=O)[O-])c1 c1(C(CNCC(C(=O)NC)COC)O)ccc(Cl)cc1F c1(COC(C(=Cc2ccccn2)C)=O)ccc(F)cc1N C(c1cccnc1)=CC(=O)NCCC1CCCN(C(=O)CC2(C(F)F)CC2)C1 C1(CC(=O)NC2(CF)CCN(C(c3snc(Cl)c3Cl)=O)C2)CCCC(F)(F)C1 CC(C)C(C)CC(=O)NCCc1ocnc1CNC(=O)C(C)n1cccn1 N1(CCN(CC(=O)N(CCC(C)C)C)CCO)CCOC(C(N)=O)C1 N1(C(c2c(CC)con2)=O)C2CCC1CN(C(=O)C#CC1(C)CCCO1)CC2 CCCCCCC(CC)C(=O)N1CCN(Cc2cccc3c2OCCO3)CC1C C(=O)(CCCCCN(C(=O)CC)CCNC(=O)CCC1CC1(C)C)OC(C)(C)C C(=O)(C(C)(C)CS(N)(=O)=O)N1CCCC(C(=O)NC2(C)COC2)C1 c1(OCC)cc(C(=O)Nc2ccc(O)cc2O)c(-c2ccc(O)c(OC)c2)cn1 C1(NC(C(F)=CCC)=O)CN(C(c2nnsc2C)=O)CCC1O c1(CN2C3CN(c4ccnc(C(F)(F)F)n4)CC32)ccc2c(Cl)ccnc2c1 C(=O)(CCCC1CCCC1)N(C1C(CC)CC1)C=O.CC(CCc1cn[nH]c1)n1cccn1 C1(NC(c2c(OC)c(Cl)sc2)=O)CCC12CN(C(c1ccc(N)cn1)=O)C2 C1(n2cc(CNC(=O)OC)nn2)CCCN(C(=O)CCCCF)CC1 CCCCCCCCCC=CC(N1CC2CCC(C1)N2C(C1(C)CCC1)=O)=O CC1(C)C(n2cc(C(C3CC3)C(N)=O)nn2)c2ccccc2N1C(c1ns[nH]c1=O)=O c1(C(N2C(CNC(CCC(C)OCC)=O)COCC2)=O)ccc(N)c(Cl)c1 c1(C(=O)NCC2C(NC(Cc3c(C)noc3)=O)CC2)nc2c(s1)CN(C)CC2 N1(C(CS(CC)(=O)=O)=O)CCOC2(CCN(C(C3CC(F)C(=O)N3)=O)C2)C1 N1(C(CC#N)=O)CC2CCC(C1)C(NC(C13CCCCC1C3(F)F)=O)C2 C1(CCNC(C(CC)C)=O)CCCN(C(=O)CC2CC3CCC2O3)C1 N1(C(C2CCC(C)CC2)=O)CCC2(CCOCC2)C(CNC(C2(O)COC2)=O)C1 Cc1cc2nccnc2cc1C(=O)NCCC(C)NC(C1CCC(F)(F)C1)=O C1(NC(c2c(C)nn[nH]2)=O)CCCCCC1NC(c1cnco1)=O Cc1ncc(Cl)c(C(=O)NC2CCN(C(=O)CCOCC3CCCO3)C23CC3)n1 N1(C(C2N(C(CC3C(C)(C)C3(C)C)=O)C3CCC2C3)=O)CCN2C(=O)NCC2C1 C1(NC2CCN(C(C(=O)NC(CC)C)C3CC3(C)C)C2)CCN(S(C)(=O)=O)CC1 Cn1nccc1C(=O)NCC1CCC(NC(C2(C(F)(F)F)CCCC2)=O)C1 c1(C(=O)NC2CC(CNC(c3c(C)n(C)nc3)=O)C2)cc(Cl)cc2c1OCC2 C1(C(N2CCC(CNC(c3ccnc(OC4CCC4)c3)=O)C2)=O)CCC(F)(F)C1 C#CCC(C)(CC)C(=O)NC(CNC(c1cc(NC(C)=O)ccc1Cl)=O)C(C)C N1(C(C=CCN(C)C(C2CN3CCC2C3)=O)=O)CCCCC1CCCO N=c1ccc(C(N2CCCC2c2ccc(Br)s2)=O)n[nH]1 C(CCC(C)C)(C(=O)NCCN1CC=CCC1)NC(C(C)OCCCC)=O C(CN=c1[nH]c(=NCC(C)(C)CCC#N)[nH]c2c1CCCCC2)SCC C(=O)(CCCCCCCCC1CC1)NC1C(NC(CNC(=O)Cn2cncn2)=O)C1 c1(C(N)=O)nccnc1C(=O)NCC1(CNC(c2ccccc2F)=O)CCC1 C1(CNC(=O)CCC2CCOC2)CCCCN1C(=O)CCCc1cccc(Cl)c1 Cc1cc(C(=O)NCC(O)CNC(C2CCCC2(C)C)=O)ccc1-n1cncn1 N1(C(C=C(C)CNC(c2c[nH]nc2Cl)=O)=O)CC2C(C1)C2(F)F Cc1ccc(C(=O)NCCNCC(C)C2CCC2)cc1Br CC(C)CCC(F)C(=O)NCC1CCCCC1C(=O)NCC1CC2CCC2C1 N1(C(C2CC(OCC)C2)C(=O)NCc2conc2C)CCCCC12CCC2 c1(C(=O)NC2C(C)CN(C(=O)CC3(CO)CCCCC3)C2)cc2n(n1)CCCO2 N1(C(c2cnn(CCCC)c2C)=O)CC(NC(c2coc(Cl)n2)=O)C2(CC2)C1 c1(C2(C(=O)NC(CCNC(C3CN(C(C)=O)C3)=O)CO)CC2)ccnc(Cl)c1 c1(C(N2C3(C(=O)NCCc4nc(CC)[nH]n4)CC3CC2)=O)cc(C)ccc1C Cc1nc(C)c(CC(N2CC=CC2CNC(=O)C(C)c2cccs2)=O)c(O)n1 c1(OC)ccc(C(=O)NCCC2CCCN2C(=O)C=C2C3CC4C(C3)C24)c(F)n1 C1(NC(CCCOCCC)=O)CCCN(C(c2cscc2Cl)=O)C1 C(=O)(CC(C(F)F)NC(C1CC2(CC2)CO1)=O)NCCNC(COC)=O C1(C(=O)NC23CCC(CNC(=O)C(F)F)(C2)OC3)Cc2ccccc2O1 C1(NC(CC=CC(C)(C)C)=O)CCCC1NC(c1cc(C2CC2)no1)=O N1(C(c2c(C)scc2)=O)CCCN(C(C2CC2(C)Br)=O)CC1 C(=O)(C1=CC(C)(C)C1)N(C(C)CNC(=O)C(c1cccc(N)c1)O)C C12(NC(=O)Cc3ccoc3)CCN(C(=O)CC3CCCCC3)CC1C2 N1(C(c2ccncc2F)=O)CCC2(C=C(C(=O)N3CCC(CF)CC3)C2)C1 c1(CC(=O)NC(CCOC)CNC(c2ccnn2C)=O)cccc2ccccc12 c1(C(=O)NCCCCCNC(CC2(OC)CC2)=O)cccc2ccsc12 C=CC(C)CC(=O)N1CC(c2ocnc2CNC(=O)C(C)CF)C1 C(=O)(CCC(C)(C)C#N)N1C(CCNC(C2ON=C(C)C2)=O)CCCC1 CC1C(=O)NCCN1C(=O)Cc1ccc(NC(C2COC(C)C2)=O)cc1 c1(N2CC(C)OCC(C)(C)C2)nc(=NCC2(Cl)CC2(F)F)[nH]c2c1CSC2 N1(C(C2(CCC=C)CC2)=O)CC=C(CNC(c2csnc2C)=O)CC1 C(CN=c1[nH]c(=NCc2cccc3[nH]ncc23)c2[nH]ccc2[nH]1)C1(C)CC1(F)Cl c1(C(=O)NC2C(CC)NCC2)csc(Cl)c1Br C(C(CNC(=O)C(C)Cc1cnn(C)c1)C(F)(F)F)NC(CCC(=C)C)=O Cc1cc(F)c(Br)cc1C(=O)NCC#CCNC(c1ccccc1O)=O c1(C(N2C(CNC(C3N(S(C)(=O)=O)CCCC3)=O)C=CC2)=O)ccc(O)nc1Cl c1(C(N2CC(O)(C(C)NC(C(CC)C)=O)C2)=O)ccc2c(c1)CCCS2 c1(C(=O)NCC2(OC)CN(C(C3(OC)CC3)=O)C2)cc(F)c(C)c(N)c1F c1(C(N2CCC(F)(CNC(C(C3CC3)OCC)=O)C2)=O)ncc(C)cc1C C1(CNC(C2COCCO2)=O)CC2CCCC(C1)N2C(c1ccc(O)nn1)=O c1(C(=O)OC)cncc(NC(C2CCC(CCO)CC2)=O)n1 C(C(=O)NOC1CCCN(CC)C1)(C1CCC1)NC(Cn1ncc(CC)c1)=O C1(C(N)=O)CC(NC(c2ccccc2Oc2cccnc2)=O)C12CCC2 c1(NC(c2cccc(C(F)F)n2)=O)ccc(F)cn1 Cn1nnc2c1CC(C(=O)NC1CC1CNC(C1CCC3(CC1)CC3)=O)CC2 O=C(N=c1[nH]ncn1-c1ccccc1)NCc1ccccc1-c1ccc(F)cc1 C1(C(=O)OCC)CCN(C(=O)C(=O)NC(c2ccc(Cl)c(F)c2)C)C(C)C1 c1(C(N2C3CN(C(COCCCCCCCC)=O)C(C3)C2)=O)cc(F)cc(Cl)c1N C1(CNCC2(F)CN(C(C(C)OCCOC)=O)C2)CCCC12CC2 N1(CC(CCC)NS(=O)(=O)CC)CCCC(CC(=O)OC)CC1 C1(C(=O)NC2(CC=C)CC2)CCN(C(=O)CC(F)(F)F)CC1(C)C C1(CC(=O)NC(CN(C(C2(COC)CC=CC2)=O)C)(C)C)CC2CCC1CC2 Cc1cc(C)c(C(=O)NC(C)C(C)NC(=O)CCc2ccc(O)c(F)c2)c(=O)o1 C=CC(CCC)CC(=O)NCC1(OC)CCN(C(=O)C(CCSC)NC=O)C1 Cc1cnc2cccc(CN3CCC(OCC4CCCCC4)C3)n12.N12CC(CC1)O2 CCCC(CC(=O)N1CCC(NC(C)=O)C1)NC(c1c[nH]c(C)c1)=O c1(C(N(CCCNC(CC(C(CC)C)O)=O)C)=O)cc(=O)c2ccc(O)cc2o1 CCS(=O)CC(=O)NCC(C)(C1CC1)NC(=O)CCc1ccc(OC)nc1 c1(SC)cc(C(N2CCC(NC(=O)Cc3nnc(O)s3)C(C)C2)=O)ccc1Cl C(C(C)(C)CCCO)N.c1(Sc2n(C(CC)C)nnn2)ccc(OC(F)F)nc1C=O Cc1cc(C(=O)NCCC2COCCN2C(C2CSCC(=O)N2)=O)sc1C N1(C(c2n(CC)nnc2)=O)CCC(C)(CC(=O)NC(C)CN(C)C)C1 C(CC(=O)NC1(C2CCCN2C(c2cnc(SC)nc2)=O)CC1)(C(C)C)OCC CCC(C(=O)NCCC(=O)OC(C)C)C(F)(F)F.C1C(=O)N1 N1(C(C(COC)N(C)C)=O)CCC(F)(CNC(c2sc(C)cc2OC)=O)C1 c1(C(N2CCC(C)C(NC(=O)CCCn3cccn3)C2)C)ccc(F)c(F)c1 C(CCOC)(C(=O)OC)NC(c1n(C(CC)(C)C)nnn1)c1cocn1.C1CO1 N1(C(C(CC=C)CC(F)F)=O)CCCC2(CCCN2C(C2CCNC2=O)=O)C1 N1(C(CCCOC(C)=O)=O)CCCC2(CC(NC(c3cnn(C)c3Cl)=O)CO2)C1 c1(C(=O)NCCCN(C(CC=C(C)C)=O)C)cc(Br)c(C)cc1F N1(C(COCCSC)=O)CCS(=O)(=O)C(CCNC(=O)C(=Cc2cccs2)C)C1 N1(C(C=Cc2ccc(SC)s2)=O)CCN(C)C(CNC(C2CC2C)=O)C1 C(C(CNC(=O)CCCn1cccn1)C(F)(F)F)NC(C(c1cnn(C)c1)C)=O C(=O)(CC(C)(C(F)F)N(C)C)N(CCNC(c1nc(C)[nH]c1C(F)(F)F)=O)CC N1(C(C(C=C=C)C)=O)CC(NC(=O)CCc2nc(C3CCCC3)no2)C(C)(C)C1 N1(C(CC2C(NC(CNC(CCC)=O)=O)CCC2)=O)CCCCC1C(C)(C)O c1(OC)noc(C)c1C(N1CCN(C(=O)C(C)OCCN(C)C)CC1)=O c1(C(=O)NCCC2N(C(c3cnc(C)s3)=O)CCSC2)ccc(C(C)C)nc1O C1(CNC(CC(C)O)=O)CN(C(c2ccn3cncc3c2)=O)CC12CCC2 c1(C(N2CCC(C)C(CNC(c3ccc[nH]3)=O)C2)=O)csc2cc(Cl)cnc12 c1(OC)cc(Br)ccc1S(=O)(=O)N1CCCC(NC(c2ccccc2)(C)C)CC1 c1(C(N(CCCNC(C2(CC)CC2)=O)CC)=O)cc(C#N)c[nH]1 C(=O)(C(CO)C(C)(C)C)NC(CCCNC(c1c(Cl)cn(C)n1)=O)c1ccccc1 N1(C(c2n(CC)ncc2Cl)=O)CCN(C(C2CCCCC2)=O)C(CS(C)(=O)=O)C1 C1(NC(C23OCC(C)(C2)C3)=O)CC12CCN(C(C1CCCCN1C(N)=O)=O)CC2 CCC(C)(C)C(=O)C(=O)N1CC(C(O)C(=O)NCC(c2ccccc2)F)C1 CC1(C(=O)NCC2(CC(=O)NCC3(CO)CCOC3)CC2)COCCO1 c1(C(=O)NCCC2CCC(NC(c3[nH]cc(C)c3)=O)C2)n[nH]c2c1CC(C)CC2 N1(C(=O)C(c2cccnc2)O)CC2CC(C1)CN(C(C1C=CCC1)=O)C2 c1(C(N(C(CNC(COc2c(C)c(Cl)ccc2)=O)C)C)=O)ccc(S(C)(=O)=O)[nH]1 c1(C(=O)NCC2C(NC(C3N(S(CCC)(=O)=O)CCC3)=O)CC2)cnn(C)c1F C(=O)(CC(C)(C)CCC)NCCCN(C(C(CCC)CC1CCCC1)=O)C(C)C N1(C(C=C(C)C2CC2)=O)CCC2CCN(C(c3ccc(C4CC4)cn3)=O)CC12 C(=O)(C(O)C(C(C)C)OC)N1CC(C(=O)N(C)CC2CCCCCC2)(SC)C1 Cc1nc(Cl)ccc1C(=O)NCC(C)CN(c1cc(O)ncn1)C C(c1cccs1)=C(C)C(=O)NCC(C)(C1CC1)NC(=O)CCC1CCOC1 CC(CF)C(=O)NC1CCC(CCNC(c2cnnn2C)=O)C1 N(C(=NCc1ncnn1C(C)(C)C)NC1CCCC1)Cc1n(C(C)C)ncn1 N1(C(c2nc3n(c2Br)CCC3)=O)CCCC2(C1)CN(C(C1(F)CCC1)=O)C2 C1(CC(=O)N(C)CC2CC2(C)C)CC2(C1)CN(C(C1(C)CC3(CCC3)C1)=O)C2 C(=O)(CCCN(C)C1CC1)N(C1CCN(Cc2cc(-c3cccs3)[nH]n2)C1)CC N1(C(c2c[nH]c(=NC)o2)=O)CC2(CCC(CNC(C3CCCOC3)=O)O2)C1 c1(N(CCNC(C(CC)CCOC)=O)C)cc(C)nc(O)c1C(=O)OC(C)(C)C C1(C(=O)NC(c2nncs2)C)CCN(C(c2n[nH]c(O)n2)=O)C1 C1(N(CC#C)C(C2CCC(CC)O2)=O)CCN(C(c2ccnc(C)n2)=O)CC1 c1(C(=O)NCCCN(C(COCCOCCOCC#C)=O)C2CC2)cc[nH]c1C c1(C(=O)NC(C(C)NC(c2cccc(CC=C)c2)=O)C)ccc(OC)cc1C n1(CC#C)cccc(CC(=O)NC2CC(C(=O)O)C23CCC3)c1=O C1(N(C)C(c2c[nH]cc(Br)c2=N)=O)CC2CCC(C1)N2C(c1ccc(F)o1)=O N1(C(C(C)OCC=C)=O)CCC(F)C(NC(=O)C=C(C)c2ccccc2)C1 c1(C(=O)NCC(CCOC)NC(CNC(CCC)=O)=O)ccc(OC(F)F)cn1 C1(NC(=O)CCc2ccc(O)nc2)CN(C(c2nc(Cl)c(Cl)s2)=O)CCC1CO c1(C(=O)NC2CCCC(NC(c3cc(C4C(C)C4)on3)=O)C2)cccc(C#N)c1 c1(OC)ccc(C(=O)NC(C2CN(C(c3ccccc3C3CC3)=O)C2)C)c(Cl)n1 C1(CC)CCCN(C(c2cc(O)ncn2)=O)C1C(=O)NCC(C)CC(C)C S(=O)(=O)(c1cc(Br)ccn1)NC(CCc1ccc(C(=O)O)cc1)=O N1(CC(C)CNC(=O)NC(C)CC2CCCO2)CCOC1=O N1(C(COCC)=O)CCC2(CCC(C(=O)NCC3(O)CC3)O2)CC1 C1(CC(=O)NCCCn2c(C)ncc2)CCCN(C(=O)C(C)(O)C2CCC2)C1 C(=O)(C(CC)C(F)(F)F)NCCCN(C(C1C(CC)N(C)CC1)=O)CC C(CN=c1cc(C)c(S(=O)(=O)N(C)CC2CCCOC2)c[nH]1)N(C)CC c1(C(N2CC(N(C(c3c(C)ccnc3Cl)=O)C)C2)=O)cnc2[nH]cnc2c1 c1(C(N2CC3CC(NC(c4c(COC)cco4)=O)C3C2)=O)ccc2cc[nH]c2n1 Cc1cc(C(N2CCOCC2CNC(C2CC2CF)=O)=O)n(C)n1 c1(C(N(CCN(C(C)C)C(c2cnsc2)=O)C)=O)cc(N)c(Cl)c(O)c1 N1(C(CCN(CCC)C)=O)CCC(CO)(NC(C2C(CN=[N+]=[N-])C2(C)C)=O)C1 c1(CCNC(C=C(CC)C)=O)ccc(N2CCN(C(c3cnc[nH]3)=O)CC2)cc1 N1(C(c2ccc(OCOC)cc2)=O)C2CCC1CN(C(c1cccnn1)=O)CC2 C1(CNC(C(C)SC)=O)CC2CCC1N(C(=O)CC(C(F)F)n1ccnc1)C2 c1(C(=O)NCC(CCOC)NC(C2(COC)CC2)=O)cc2cccc(C)c2o1 Cc1noc(C(F)(F)F)c1C(=O)NCC1(CNC(C2CC2F)=O)CCCC1 CC1CN(C(C2(O)CCCCCC2)=O)CC(C)N(C(=O)CN(C)C2CC2)C1 C1(CNC(Cn2ccc(C)n2)=O)CC2CCC1N2C(c1cc(=N)[nH]n1C)=O C1(NC(CCC)=O)CCC(CNC(=O)CCCc2ccc(C)s2)C1 Nc1ccc(C(N2CCCCC(NC(=O)CCNC(N)=O)C2)=O)c2cccnc12 c1(CCC(=O)NCC(C)N(C(CC2ON=C(C)C2)=O)C)ccc(Cl)c(F)c1 N1(C(c2nc(CC)oc2C)=O)CCN2C(=O)C(NC(c3ncn(C)n3)=O)CC2C1 c1(C(N2CCCC(CN(C(C(C)SC)=O)C)C2)=O)c[nH]cc(Br)c1=N c1(C(=O)NC(CC(C)NC(C2CC(=C)C2)=O)C)ncccc1NC(C)=O C(=O)(C(C)C(C)(F)F)NCC(CC)(CC)NC(c1ccc([N+](=O)[O-])s1)=O C(=O)(CC(O)CCSC)NCCCNC(C1C(OC)CC1)=O C1(N(C(=O)CN2CCSCC2)C)CC2CCC(C1)N2C(=O)C(C)(C)S(C)(=O)=O C1(NC(CC2CC(OC)C2(C)C)=O)CC2(C1)CC(NC(C1CN(C)C1)=O)C2 c1(OC)cccc(C(=O)NCC2(C(C)(C)C)CCN(C(=O)C(CO)N(C)C)C2)c1 c1(Cc2cn(C)nc2)ccc(CCNC(=O)NC2(c3ccno3)CCC2)cc1 N1(C(CC(CCC)NC(c2ccc(NC)cn2)=O)=O)CCn2ccnc2C1 Cc1n[nH]c(C)c1C(=O)NC1C=CCN(C(c2[nH]ccc2C2CC2)=O)C1 Cc1nc(C)n(O)c1C(=O)NCC(C)(F)CNC(C1CC(Cl)(Cl)C1)=O N1(C(c2c(CCN(C(C(C)CN(C)C)=O)C3CC3)c[nH]n2)=O)CCCCCC1C C1(NC(CCN(S(C)(=O)=O)C)=O)CCCCC1CNC(c1ccc(F)cn1)=O Cc1nc(N2CCCC(NC(=O)CCNC(c3ccco3)=O)CC2)c2ccsc2n1 N1(C(c2cccc(OC)n2)=O)CCC(C2(NC(=O)C(C)C(C)O)CC2)C1 Cn1cc(C(F)=CC(=O)NC2CC(C)(NC(c3cc(O)ccc3Cl)=O)C2)cn1 N1(C(C(CCC)OCC)=O)CCN(C(=O)CCn2ccnc2C)C2COCC12 CC(C)(F)C(C)(F)C(=O)N1CCCC(NC(C2(c3ccccc3C#N)CC2)=O)C1 C1(NC(C2CCOC2)=O)CCN(C(=O)Cc2cncnc2)C1c1ccccc1 c1(C(=O)NCC2(CNC(c3cc(O)ncc3Br)=O)COC2)cc(Cl)cc(Cl)c1Cl c1(OCC)ccc(CCC(=O)NCCCN(C)C(C2SCCC2C)=O)cc1 C1(CC#C)(C(=O)NCSc2ccc(Cl)cc2)CCN(S(=O)(=O)CC(=O)OC)CC1 O=C1CCOC(C(N2CC(N3CCN(C(=O)CN4CCCNC4=O)CC3)C2)=O)C1 c1(NCCC(C)C)cc(=NCC(Cc2ccc(Cl)cc2)CO)[nH]c(C(F)(F)F)n1 C#CC1(C(=O)NCC(C)(O)CC)CN(C(C23CCC(C2)C3)=O)C1 Cc1c(CC(N2CC(F)CC2C(=O)NCC(c2nncn2C)C)=O)cnn1C CCC(C)N=c1[nH]c(=NCc2n[nH]c(=N)s2)c2c(F)cccc2[nH]1 c1(C(=O)NC2CC2CNC(c2cnc(Cl)[nH]2)=O)ccc2nccnc2c1 Cc1cc(F)cnc1C(=O)NC1CC1CNC(c1cccc(C2CC2)c1F)=O c1(C(N2CC(CC)C(C(N3CCOC(C(C)(C)C)C3)=O)C2)=O)cccc(O)c1C c1(C(=O)NCC(CC=C)NC(=O)C(C2CC2)N(C)C)ccc2cccnc2c1N C=CCCCCCC(=O)NCC1CN(C)CCN1C(c1cncc(Cl)c1C)=O CCCC(CC)C(=O)N1CC(F)CC1CC(=O)NCc1ncn(C)n1 N1(C(c2c(C(C)C)n[nH]c2)=O)CC2CCC(C1)N2C(C1CC(=O)CCO1)=O CC(C)(O)C#CC(=O)N1CC=CC1(C)C(=O)NC1CCOC(C)(C)C1 Cc1ncc2cc(C(N3CCC(C)(C)CC3CNC(=O)C(F)(F)F)=O)ccn12 C1(C)(CNC(c2n(CC#C)cnn2)=O)CCN(C(c2cncc(F)c2)=O)C1 n1(CC)ccc(=NC(=O)C2CCN(C(=O)CN3CCSCC3)CCO2)[nH]1 C(=O)(CCC(C)(C)F)N(C(C)CN(C)C(C1(CNC(=O)OC(C)(C)C)CC1)=O)C C1(CC)(CNC(=O)C(CCC2CCC2)NC(C2CC(F)C(=O)N2)=O)CCC(=O)N1 C=CCC(CC(C)C)C(=O)N(CC(N1CCCC1CCC(C)C)=O)C1CC1 CCCC(CNC(C1(C)CCNC1=O)=O)C(=O)NCCc1cnccc1C C1(CNC(c2c(C)ccnn2)=O)CC12CCN(C(=O)C=Cc1ncc[nH]1)CC2 N1(CC)CCOCC1CN(C(=O)CC1CCN(C(=O)C=C(C)C)C1)C c1(C(C)NC(=O)CCNC(C2C3COCC23)=O)ccccc1F N1(C(CCN(C)CC)=O)CC2(CC2)CC1CC(=O)NCc1ccnc(C)n1 CCCCCCCCC(F)C(=O)N1CCC1CNC(=O)C(C)(C)CC(=O)OC C(=O)(C(C)CC(F)F)NC(CNC(c1c(C)onc1-c1ccncc1)=O)C C(=O)(C(C(C)(C)C)NC(C1CC(OC)C1)=O)Nc1ccc(OCC)nc1 c1(CC)oc(C)cc1C(=O)NC(C)(CO)C(=O)N1CCC(C(C)(C)O)C1 c1(C(=O)NC2CC3CN(C(CSC(C)(C)C)=O)C2C3)cnc2[nH]cnc2c1 CC1(NC(c2cnc[nH]2)=O)CCN(C(C2CCCN2N=O)=O)CC1 N1(C(C(C)OCCC#C)=O)CCC(O)(CNC(c2cn(CC)cn2)=O)C1 CC(C(=O)NCCNC(=O)Cc1ccc(O)cn1)(C(F)F)c1ccccc1 C1(C(=O)NCC(C2CCC2)NC(C(CC=C)(C)C)=O)CCCC2(CCC2)C1 c1(C(=O)NC(C)(C)CNC(=O)C=CC(=O)NC2CC2)ncn2c1CCCC2 c1(C(N2CC(CNC(C3(CSC)CC3)=O)C(O)C2)=O)c(C)cc(C)cc1N N1(CC(=O)NCC2(CCNC(C3(F)CCS(=O)(=O)C3)=O)CC2)CCS(=O)(=O)CC1 CC1C2=C(C(=O)N1C)C(c1cc3sccc3n1C(C)(C)C)NC(=O)N2CC1CC1 c1(CC)nccnc1C(N1CCC(C)(NC(C2COC(=O)O2)=O)C1)=O C12(C(N(C)CC3(OCC)CCC3)=O)CCCC1CCN2C(=O)Cc1cc(C)[nH]n1 c1(C(N2CCN(C(c3c[nH]ccc3=O)=O)C3CC23)=O)cccc(F)c1F O=C(C1=CCN(C(C2CC=CC2)=O)CC1)NC1CCOC1 N1(C(C(C)CF)=O)CC2CC1CN(C(=O)CSCc1nc3ccccc3[nH]1)C2 c1(C(=O)OC)ccccc1C(N1CC2CC2(CNC(c2cc(C)ncn2)=O)C1)=O c1(C(N2C(CNC(CCC)=O)CC(C)(C)C2)=O)cc2cc(Cl)ccn2n1 c1(C(C)C)ccc(C(N2CC(F)CC2CNC(=O)CS(=O)(=O)N(C)C)=O)nc1 C(=O)(CC(C)(C)C(=O)N1CC2(CCC2NC(=O)COCC2CCC2)C1)OCC N1(C(C2(CCNC(C3CCCCC3F)=O)CC2)=O)CCCN(C2CCC2)CC1 N1(C(c2c(C)nn[nH]2)=O)CCN(C(c2ccc(I)c(Br)c2)=O)CC1CO C(=O)(C#CC(C)(C)C)NC(c1ccc(C(N2CC(OC)C(OC)C2)=O)cc1)C CC1(C)C(NC(c2csc3nnsc23)=O)CCN1C(c1ncccc1Cl)=O N1(C(c2ccc(C)nn2)=O)CC(NC(c2cn(CCCC#N)nn2)=O)CC(O)C1 c1(C(=O)NC(C(=O)OC)C(C)C)ccc(CN(C)C)cc1C.C1(=O)CO1 C1(NC(N2C(COC)COCC2)=O)COCCN(c2nc(C)cs2)C1 N1(CC(=O)NC(CN(C(c2oc(C(F)F)cc2C)=O)CC)C)CCCC(CO)C1 N1(C(C2C(OCC)CC2)=O)CCN(C(c2cccc(Cl)c2Cl)=O)C2CCC12 C1(NC(C(C)SCCCC)=O)CCN(C(=O)C(c2cn(C)nc2C)O)CC1O c1(C(NOCCC=C)=O)ccc(CNC(C2(C#N)CCOC2)=O)cn1 CC1(C)C(NC(c2nocc2Cl)=O)CCN1C(=O)CC1CCCCC12CC2 C(=O)(C1=CC2CCCC12)N1CCC(F)(CNC(C=CCOCCOC)=O)CC1 c1(NC(C)=O)ccc2c(CNC3CCSc4c(F)cccc43)cc(=O)oc2c1 N1(C(C(C)SCC)=O)C2CCCC1CN(C(=O)C(C(C)C)OCC(C)C)C2 c1(CCC(=O)NCC(CN(C(CC2(C=C)CCC2)=O)C)O)c(F)cccc1F N1(C(C(CC=C)NC(C)=O)=O)CCC2(CC2)CC1C(N1CC2C=CC1CC2)=O Cc1cc(O)c(-c2noc(C3CCN(c4ccc5nncn5n4)CC3)n2)cc1Cl C(=O)(CCS(=O)(=O)Cc1cccc(C)c1)N1CC2C(CNC(C(CC#C)C)=O)C2C1 C1(NC(C(CC2CCC2)NC(=O)CC2CCCSC2)=O)CCCC(O)C1 c1(C(=O)NCCN(C(C2C(C)CCS2)=O)C2CC2)ccc(S(=O)(=O)CCO)cc1 N1(NC(NCC(C=C)(C)C)=NCCOC)CCC2C(C1)C2(F)F CC(CC(=O)NC(C)(C)CNC(c1ccc(C#N)nc1O)=O)CC(C)(C)C C(=O)(C1CCCc2c1ncn2C)N(CC(C)Nc1cc(C(C)(C)C)ncn1)C C1(C(N2C(C#C)CC2)=O)(CNC(=O)CCc2nncs2)CC2(CC2)C1 C(CNC(c1ccc(CC2CC2)cc1)=O)(C(C)(C)C)NC(CC(C)SC)=O CCC(CC)C(C)C(=O)N(C(CC)CC(=O)NCCC1CC(C)=NO1)C N1(C(C(C2CCCOC2)NC)=O)CC2COCC2C1 C1(NC(C=CC(C)(C)SC)=O)CCCC1(C)NC(c1ccsc1C)=O C1(C2CCCN(C(=O)Cc3ccco3)C2)(NC(=O)Cn2cc(F)ccc2=O)CC1 N12CCOC(C1)CNC2=O.C12(NC(C3(CC)CCC3)=O)CC(C(F)(F)F)(C1)C2 C1(C(N(CC(C)C(=O)NC(C2CC2)C2CC2)C)=O)C2CCC(F)C12 C1(CSC)CCCN(C(=NC(C)CC2CCCCC2)NCC2CCOC2)C1 C1(CNC(C2CCC2C(F)F)=O)CCN(C(=O)C(C2CCOCC2)F)CC1(F)F C1(CN(C)C(C2CC(O)C2)=O)CCCCN1C(=O)C=Cc1cc(C(=O)OC)co1 c1(NC(c2n[nH]c(C)c2C)c2n(CCCOC)nnn2)cn(C)nc1C N1(C(c2cc(C)ncc2)=O)CCC(CNC(C2OC(C)CC2C)=O)CC1C C1(CC)(NC(c2cc(CO)oc2C)=O)CCN(C(C2CCC(C)(C)CO2)=O)CC1 C1(NC(C2(CCC)CC(=O)C2)=O)CCCC(C(=O)NC(CC)C(C)(C)O)C1 N1(C(CN(CCC#C)C)=O)CCCC(CO)(CNC(C2CCC(=O)N(C)C2)=O)C1 c1(C(N(CC)CC2CCCN2C(=O)CCCC(C)C)=O)nn(C)c2c1CSCC2 C1(O)(C(N2CC(CC=C)(NC(=O)CCC3C(=O)NN=C3C)C2)=O)CCCCC1 c1(C(=O)NCC2CN(C(CC3CC(C)C3)=O)CC2O)ccn2ccnc2c1 N1(C(c2n(C)nnc2Br)=O)CCC(O)(CCNC(c2cc[nH]c2)=O)CC1 C1(O)(n2cc(SC(C)(C)C(=O)O)nn2)CCN(C(C2CCC(F)CC2)=O)CC1 c1(C(N2CCC(CN(C(Cc3c(C)n[nH]c3)=O)C)C2)=O)ncn2cc(Cl)ccc12 C1(NC(C2(N(C)C)CC2)=O)CCN(C(c2cncc(O)c2Cl)=O)CC1CO c1(CC(=O)NCC2CN(C(C3CCC(C)(CC)O3)=O)C(C)C2)cc(C)cc(F)c1 O=C(CCN(CCCO)C(c1cnco1)=O)NCC1CC1 Cc1ccc(F)c(C(N2CC(NC(C3CC4CC4C3)=O)CC(F)C2)=O)c1Cl CC(C)CC(C)(CNC(C1(F)C(C)(C)C1(C)C)=O)NC(c1cc(F)cc(F)c1)=O C1(C(=O)NCC2(NC(c3cccc(SCC)c3)=O)CC2)COCCN1C=O N1(C(N2CCC(Oc3ccc4c(c3)OCO4)CC2)=O)CCC(C2CC2(F)F)CC1 c1(NC(CCC2N(C(C(CCC)N(C)C)=O)CCCC2)=O)cccn(CC)c1=O N1(C(C2(SCC)CC2)=O)CCC(CF)(NC(=O)C(C)C2CCCC2)C1 C1(n2cc(-c3c(F)ccc(C(=O)OC)c3)nn2)CN(C(COCC)=O)CC1C1CC1 C1(CNC(C(COC)(C)OC)=O)CCn2cncc2C1.C1(=O)CCCN1 c1(C(=O)NC2CCC(NC(C3C(OC)CC3)=O)CC2)cc2ccc(SC)cc2[nH]1 Cn1nc(C(=O)NC2C3CC2N(C(c2c[nH]c(N)c2)=O)C3)c2c1CCC2 C1(COC)(NC(=O)C(C2CCCO2)C2CC2)CCN(C(=O)CN2CCCC2)CC1 C1(C(N2C(C(=O)NCCC(C)O)(COC)C=CC2)=O)OCCCC1(C)C S(=O)(=O)(CC(=O)N1CC(O)(CCNC(c2nccnc2C(=O)OC)=O)C1)NCC C(C(C(F)(F)F)N1CCN(C(=O)CCc2ccsc2)CC1)NC(C(C=C)O)=O C(=O)(C(F)C(C)(C)O)N(CCCNC(C1CC(=C(F)F)C1)=O)CC N1(C(COCCCCC)=O)CCC(O)(C(C)NC(=O)C(C)OCC)C1 O=C(CCC(F)(F)C(F)(F)F)NC1(CO)CN(C(=O)C(C2CCCCCC2)O)C1 Cc1ccc(C(C)C(N2CCC(O)(CCNC(=O)C=Cc3cc[nH]n3)C2)=O)cc1 C(c1cc(F)cc(F)c1)=CC(=O)NC1(COC)CCN(C(C(C(CC)C)O)=O)C1 N1(C(C(C)OCC=C)=O)C2CCC1CC(CNC(=O)CCc1ccnc(C)n1)C2 C(=O)(C1=CC(O)C(O)C(O)C1)N1CCC=C(C(=O)Nc2c(C)ncc(F)c2)C1 c1(C(=O)NC(c2cn(Cc3ccc(Cl)c(Cl)c3)nn2)C)cn(C)ccc1=O c1(OC)coc(C(N2CCCC(C(C)NC(=O)C=CC3CC3)C2)=O)cc1=O C(=O)(CC(=O)NCCCCC1CN(C(C23CSCC2C3)=O)C1)NCC C#Cc1cnn(C)c1C(=O)NC1CC(NC(c2cnc(NC)cn2)=O)CC1O c1nnnn1CC(F)(F)F.C(C(CNC(=O)COC)CO)NC(C1(SCC)CC1)=O Cc1cc(C(N2CC(NC(=O)Cc3c[nH]ccc3=O)C(C)C2)=O)cc(C)n1 c1(C(=O)NC(CC)(C)CNC(C2CC(=O)N(C(C)C)C2)=O)cnc(C)nc1C N1(C(CCC(C)(F)F)=O)CC(NC(=O)COc2ccc(O)cc2)CC12CCC2 C(=O)(CC(CN(C)C)CC)N1C(C2(NC(CC(CC)C)=O)CC2)CCC1 c1(CNC2C(NC(c3c(OC(C)C)ccc(C)c3)=O)CC2)nnc2ccccn12 C1(C(=O)NCc2cccc(C)c2)CC2(C1)CN(C(c1ccnc(Cl)c1C)=O)C2 Cc1cc2n(n1)CCN(C(C1CC(NCc3c(Cl)cc(F)cc3Cl)C1)=O)C2 C1(CC(=O)NC(CCOC)(C)C)CCCCN1C(=O)CC1NC(=O)NC1=O CC1(CC(=O)NC2CC(CC(=O)Nn3ccnn3)C2)CCCO1 c1(CCC)ccc(OC)c(NC(=O)CC2CCN(C(c3ccc(C)nc3)=O)C2)c1 N1(C(C2(C)CC(=C)C2)=O)CC2(CCCN(C(C3CC(C4CCC4)C3)=O)C2)C1 C#CC1(C(=O)NC(C2CCN(C(c3cc(C(N)=O)c[nH]3)=O)CC2)C)CCCC1 N1(C(c2occ(C)c2)=O)CCCCC1C(C)NC(c1cc(Br)cn1C)=O N1(C(C(COC)(C)C)=O)CC(C)CN(C(c2ccc(C(F)F)cc2F)=O)C(C)C1 Cc1cnccc1C1CN(C(=O)NC2C3CCC23c2ccccc2)C1 C1(C(N2CC(CC=C)(C(N3CC(C)CC3CC)=O)C2)=O)CCOC(=O)CC1 Cc1nc(Cl)nc(N2CCCC2CNC(=O)C(=O)N)c1F.c1(NC)ccccc1 CC(C)(O)C(=O)N1CCC(C(=O)NC(C2CCOCC2)(C)C)O1 O=C(C1=COCCC1)NC(CC1CCOCC1)C(=O)Nc1cccc(CCF)c1 c1(CNC(C(n2cc(-c3cn(CCOC)nc3)nn2)C)=O)cc(Cl)c(Cl)n1C CC1(F)CCCN(C(=O)CC(CNC(=O)CN(C2CCC2)C)C2CCC2)C1 N1(C(C(CCOCC)NC(=O)C(C)CC#N)=O)CC2(CC(COC)CO2)C1 C(CC(C)(C)CC(=O)N(CCNC(=O)CN1CCOCC1=O)C1CC1)OC c1(NC(=O)OCC)ccc(C(N2CC(NC(C3CCCOC3C)=O)C2)=O)cc1 N1(C(C2CC(C)OCC2)=O)CCN(C)C(CNC(=O)CC2CC=CC2)C1 CC(C)(C)CCC(=O)N1CCCCC1Nc1nnc(C2CCC2)s1 CC1CN(C(=O)CSc2nncs2)CC1CNC(=O)CC1CCCS1(=O)=O C1(CNC(COCCC(C)C)=O)(NC(=O)CC23CCCC2C3)CCC(F)(F)CC1 C=C(CNC(c1ccnn1C)c1nnnn1CCCCCC)C1CCOCC1 C#CCCCC(=O)NCC(CC)NC(c1cc(C)c(C(=O)OC)s1)=O C1(NC(c2cc(CC)sn2)=O)(CSC)CCCN(C(=O)C(C(C)C)N(C)C)C1 c1(-n2cc(CCN(C(c3cnc(C)n3C)=O)C)nn2)ccc(C(F)(F)F)c(F)c1 N1(C(c2nn(C)c3c2CCC3)C(=O)NCCC)CCC(C#N)CC12CC2 C(CNC(=O)C(c1ccnn1C)C)(CC(F)(F)F)NC(CCCNC(=O)OC)=O N1(C(c2c(OCC)cccc2)=O)CCC2(CCN(C(=O)C(COC)OC)CC2)C1 C(=O)(C1=CCN(C(=O)COC2CCOC2)CC1)NC1(C(N)=O)CC1 N1(C(CC2(COC)CC2)=O)CC(NC(=O)CCS(N)(=O)=O)Cc2ccccc21 C(=O)(C1CCc2c[nH]nc21)NC(C1CN(C(Cc2nc(CC)sc2)=O)C1)C C1(c2cccc(Br)c2)(C(=O)NCC2C(NC(C3C(C)C3)=O)C2)CCOCC1 c1(C(=O)NCC(=O)NC2CCN(C(C)C)C2)ccccc1Br CC1CN(C(C2CC(C)(O)C2)=O)CCC1CNC(c1cnc(S)n1C)=O N1(C(c2sc(C)c(Br)c2)=O)CC(NC(c2ccnnc2S)=O)CCC1C N1(C(COCCOC)=O)CCCC(C)C1CCNC(c1nc(Cl)sc1C)=O C=CC1(C(=O)NC2CC(O)C23CCC3)CCN(C(=O)CCC(C)(F)F)CC1 C(=O)(C1CCCc2nc[nH]c21)NCc1cnn2c1CN(C(CC(C)SC)=O)CC2 C(=O)(C(CC(C)C)CC(C)C)N1CCN(CCNC(CC(CC)C2CC2)=O)CC1 C12(OC)CCC(NC(c3cnn(CCNC(c4cnc(O)o4)=O)c3)=O)(CC1)C2 n1(CC)c(C)cc(C(N2CCC(NC(c3nn[nH]c3Cl)=O)C2C)=O)c1C C1(C(=O)NC2CC(C)(NC(C(CC)OC3CCCC3)=O)C2)CC1C1CCC1 CON(CC1CCCCC1)C(=O)C1CCC(CCC(=O)OC)O1 C(C1=CCN(C(C2CNC(=O)N2C)=O)CC1)NC(c1cn(C(C)C)nn1)=O Cc1onc(C(=O)NC2CCCCC2N(C)C(c2cnc(O)s2)=O)c1[N+](=O)[O-] C12(NC(CCCNC(C)=O)=O)CC(C)(C1)OC21CN(C(=O)C(C)C(C)(C)C)C1 C1(C(=O)NC2C(NC(c3cn(C)nn3)=O)CCC2)CC(C)(C)CC(C)(C)C1 C1(C(=O)NC2(CO)CN(C(C3CC3(Cl)Cl)=O)C2)CCCN2CCCCC12 CN(CCc1ccc2c(c1)OCO2)N1CCCC(O)(c2ccccc2)C1 C1(NC(C2CC(C3CC3)C2)=O)CC2CN(C(c3nccc4cc[nH]c34)=O)CC2C1 N1(C(CCc2ccc(C)s2)=O)CC2CCC2(NC(=O)C(C(C)C)N(C)C)C1 c1(OC)ccccc1C(=O)NCC1CC2CC2N1C(c1ccoc1)=O C1(C2CCN(C(c3cnccc3Cl)=O)C2)(NC(C2CCCCC2F)=O)CC1 C1(C#CC(=O)NCC2CCC(NC(c3[nH]nnc3C3CC3)=O)CC2)(CC)COC1 C1(NC(=O)CCc2ccccc2)CCN(Cc2noc(-c3ccco3)n2)CC1 C1(NC(C2N(C(C3N(C)C(=O)OC3)=O)CCOC2)=O)CCC12CCCC2 C(=O)(C1SCc2cccnc21)N1CC(CNCc2cn(C3CCN(C)C3)nn2)C1 Cc1[nH]nc(C(=O)NC2CC(CNC(=O)C(c3ccc(F)cc3)(C)F)C2)c1C C1(C(=O)NC(C(=O)N(CC(C)SC)C)c2ccco2)C2CCC(F)C12 c1(OC)ccc(C=CC(=O)NC2CC(NC(=O)C3=COCCC3)C2)cc1O c1(NC2Cn3c(C)nnc3CC2)[nH]c(=NC2CCOCC2F)nc2sccc12 CC(CS(C)=O)C(=O)NC1CC(C)(NC(=O)COCc2nccn2C)C1 CC1(CNC(=O)C(CNC(C2CC(OC3CC3)C2)=O)SC)CCCCCC1 C1(C(C)NC(c2ccc(Br)s2)=O)CCCN(Cc2cnn(-c3ccccc3)c2)C1 CCC(C)(C)C(O)C(=O)NC12CCC(C(=O)Nc3ccc(CCF)cc3)(CC1)C2 C1(NC(C2(CC=C)CCC2)=O)CN(C(=O)C(C)(C)c2ccc(Cl)s2)CCC1CO c1(C(N2CCC(CO)C(O)C2)C(=O)NCc2ccccc2)ccc2[nH]ccc2c1 Cc1cccc(C(=O)NC(CNC(=O)CSc2nc[nH]n2)C(C)C)c1C CCC(CC)(CC)C(=O)N1CCC(NC(c2coc(C3CCC3)n2)=O)C(C)C1 c1(C(=O)NC23C(CN(C(CC(COC)C)=O)C2)C3)coc(S(=O)(=O)N(C)C)c1 c1(C(=O)NC2C3N(C(C(COC)(C)C)=O)C(CC3)C2)cnc2ccccc2n1 N1(C(CC2ON=C(C)C2)=O)CC2CC3CC2C1C3NC(c1cc(C)nnc1O)=O c1(C(=O)NCC2N(C(Cn3ncc(C)c3)=O)C3C(C2)C3)ccc(C(C)C)c(Cl)c1 C1(NC(CCN(C)CC)=O)CCCOC12CCN(C(c1cc(C)n(C)c1)=O)CC2 C1(NC(C(C)NC(C)=O)=O)CCN(C(c2csnn2)C)C1 Cc1cc2occ(C(=O)NC3COCCC3NC(=O)CC3C=CCC3)c2cc1C N(C(=NCc1cnccc1OC)NCc1nc(C2CCC2)no1)C(CC)C c1(C(N(c2ncc(-c3nc(N)cs3)cn2)C(C)C)=O)cc([N+](=O)[O-])ccc1Cl C12(C(=O)OCC)CCCC1N(C(=O)OC(C)(C)C)CCN2Cc1nn(C)cc1SC N1(C(C2C(C)(C)COC2)=O)CC2(CC2)CC1CNC(C1CC(O)C1)=O C1(CC)CC2CCC(C1)N2C(c1coc(CNC(=O)CCCN=[N+]=[N-])n1)=O c1(C(=O)Nc2cccc(CNC(C(CC=C)OC)=O)c2)ccnc(C)c1N C1(C)(C(N(C)CC2(C#N)CC2)=O)CCCN1C(=O)CC(F)(F)F CC(CN(C)C)CCC(=O)N1CC2(CCC2CNC(=O)CCCC(N)=O)C1 C1(CC(=O)NCCC(C)N(C(C2C(=C)CC2)=O)C)CCCS(=O)(=O)C1 c1(NC(=O)C(C2CCS(=O)(=O)C2)c2ccccc2)cccc(N2CCCC2)c1O c1(C(=O)NC(CC)CNC(C2(C)CCC(=O)C2)=O)sc2cncn2c1C N1(C(C(C=C)O)=O)CC2CC1CN(C(c1cc(Br)c(=O)n(O)c1)=O)C2 C(CC(O)CNC(C1CCOC1)=O)NC(c1cccs1)=O Cn1cc(Br)c2c1CCN(C(=O)Cc1ccns1)C2 CC(CCN(C)C)C(=O)NCC(C)CNC(c1cnncc1O)=O CC1(C(N2CCC(CO)(NC(c3ccc(N)c(N)n3)=O)CC2)=O)CCNC(=O)C1 CCCC(C(=O)NC1CCOCC1NC(C1(C)CCC1)=O)S(N)(=O)=O C12(C(=O)NCC3C(C)(C)C(NC(c4cnc(C5CC5)[nH]4)=O)C3)CCC(CC1)OC2 C1(NC(CC(C)(C)OC)=O)CCCC(C(=O)NCC2(C)CC(C)(C)C2)CC1 CCCC(C(=O)OC(C)C)NC(c1cc(Br)no1)c1nnnn1C(C)C N1(C(C2C(NC(c3n[nH]c(CC)c3I)=O)C3CCC2C3)=O)CCC2CCOC2C1 C(N=c1[nH]c(=NC)[nH]c(=NC(C)CN2CCCCC2=O)[nH]1)C1C(=C)C1 c1(N2CC(C(=O)NCC3CCCNC3)C(O)CC2)ncc2ccnc-2[nH]1 C(=O)(CC(C)CC(=O)N1CCC1CNC(C1CC2CCC1CC2)=O)OC C1(NC)CCC2(CCN(C(=O)C(N)CN(C)C)CC2)C1 C(CCN(C)C(C1CCN(C)C1)=O)(C(C)(C)C)NC(c1cnc(C)o1)=O c1(C(N(C(C(=O)NCCCN(CC)CC)C)C2CC2)=O)cc(Cl)n(C)n1 CCC(COC)C(=O)NCC1CC(F)(CNC(=O)CC2CCC(=O)N2C)C1 c1(C(C)NC(=O)NC(Cc2ccco2)CO)noc(C(F)F)n1 c1(OC)cc(Br)c(CC(=O)N(C)Cc2ccc(Br)cc2I)cc1F N1(C(COC)=O)CCC(NC(CCC)=O)(CNC(=O)Cc2cnccc2C)CC1 C1(c2nc(-c3cccc(F)c3)nn2-c2cccnc2)CCCc2ccccc2C1 C1(N(CCC#N)C)CCN(C(c2occc2Br)=O)CC12CC2 c1(C(N(CC(O)CN(C)C(C2(N(C)C)CCCC2)=O)C)=O)cc(N)c(F)cn1 CN1CCN(N2CCOC(NC(=O)OC(C)(C)C)C2)CC1C(F)(F)F N1(C(=O)CSC(F)F)CC2(CC(C(N3CCC3CN=[N+]=[N-])=O)CO2)C1 CCC(C)CCC(=O)NC(C)(C)CN1CCN(C(=O)C=CC(F)(F)F)CC1 C(=O)(C(CC(C)C)C(C)C)NCCn1ncc(C(=O)NC(CC)(C)CO)c1 C1(NC(c2c(CC)nn(C)c2)=O)CC(C)CN(C(c2csc(C#N)c2)=O)C1 c1(C(N2C3C(CNC(CC(CCC)O)=O)C(C3)C2)=O)cc(Cl)c(F)cc1F Cc1cc(NC(C2CC(CCNC(=O)CC(C)C(F)F)C2)=O)c(O)cc1F c1(NC(c2csc3c2CCN(Cc2cc(Br)co2)C3)=O)cc2c[nH]nc2cc1F N1(C(C(CO)OC)=O)CCC2CCCC12C(=O)NC1CC(C(C)O)C1 N1(C(C(c2ccc(Cl)cc2)C)=O)CCOC(C(=O)NCc2cncc(Br)c2)C1 C1(CNC(=O)CC2(O)CCOC2)CCCC(NC(=O)C=CC2CCOCC2)C1 N1(C(CCCC(C)=O)=O)CC2CC(NC(C3CNC(=O)C(C)(C)C3)=O)CC1C2 c1(C(N(CCN(C(C)C)C(n2ccc([N+](=O)[O-])n2)=O)C)=O)c(N)cc(F)cc1F C1(C(N2CCN(CC3(NC(CCOC(C)C)=O)CC3)CC2)=O)CCC(F)(F)CO1 C(=O)(CC(CN(C(C)(C)C(O)C(F)F)C(C)=O)CC(C)C)NCCC C1(CNC(CC2N(C)C(=O)CC2)=O)CN(C(=O)CCCN2CCCC2)CCCO1 O=C(N=c1cc2n([nH]1)CCNC2)Nc1ccsc1[N+](=O)[O-] N1(C(C2CC=CC(NC(CCc3cc(C)on3)=O)C2)=O)CC2(CCCC2)CC1C c1(C(N2C(C(C)NC(c3cn(CCCC)nn3)=O)CCC2)=O)cc(=N)[nH]c(Cl)n1 C1(C(=O)Nc2cncc(C(F)(F)F)c2)CCCN(Cc2cc(Cl)ncc2Br)CC1 N1(C(C2(NC(C)=O)CCC2)=O)CC(NC(=O)CSCc2ccc(F)cc2)C(F)C1 c1(CC(=O)NCCCN(C(=O)Cc2cnoc2)CC)cn[nH]c1 N1(C(c2c(C)cc(CC)o2)=O)CCN(C(C23CCCC2C3(F)F)=O)CC1CCO C1(NC(=O)C=Cc2ccccn2)CCN(C(C23COCC2C3)=O)CC1O c12ccc(cc1)CN(CC)CCc1cn-2nn1.C(=O)(CC(C)C)N=C(C)C(=O)O C1(C(=O)NCc2c(C)ccs2)CCC(C)N1C(c1ccc(C(N)=O)cc1)=O Cc1nc(C(N2CC=CC(NC(C3C(C)C3C)=O)C2)=O)c(C)o1 C1(Cc2nc(C)[nH]n2)CCCN(Cc2c(C)ncn2C)C1 C1(F)(CNC(C2C(C(c3ccco3)=O)CC2)=O)CC(NC(c2cccs2)=O)C1 C12(OC)CCCCC(C(=O)NC(C)CN(C(=O)C(F)(F)CN(C)C)C)(C1)C2 N1(C(c2cnn(-c3ccccc3)c2)C(=O)NCC)CCC(C)C(C(F)(F)F)C1 c1(CNCC2CCN(C(C3CCCS3)=O)C2c2cccnc2)ccc(F)cc1 N1(C2CN(C(C)=O)C2)CCN(C(=O)Cc2ccc(C(N)=O)nc2)CC1 C1(C(=O)NC(CCC(C)C)C)CCCCN(C(C2CC(F)(CF)C2)=O)C1 CC1(C(=O)NCc2ccon2)CC2CCC(C1)S2(=O)=O N1(C(c2cc(=NC)[nH]cc2)=O)CCCC2(NC(C3CCC3COC)=O)CCCC12 c1(OC)cc(C)ccc1C(=O)NCC(N1CCN(C(C23CC(F)C2C3)=O)CC1)C C1(C(N2CC3CN(C(C4(O)CCCCC4)=O)CCC23)=O)CCCC2(CCC2)O1 N1(c2ccnc(SC)n2)CC2(CC2)CC1C(=O)NCc1ccc(Cl)nc1 C1(O)(CNC(C(C)c2ccsn2)=O)CCN(C(C2(O)CCOC2)=O)CC1 C(C(C)CC(=O)N1CC(CC(C)NC(=O)CC23COC(C)(C2)C3)C1)OC c1(C(N2CCC(C)(NC(c3cc(CO)[nH]n3)=O)C2)=O)ccc(=O)n(C2CC2)c1 N1(C(c2nc(CC)sc2)=O)CCC(CC)(NC(=O)C=C2CCCCC2)CC1 Cc1cccc(C(=O)NCC2CCCC(NC(=O)C#CC3CCC3)C2)c1Cl Cc1c(C(=O)NCCCN(C(c2cccnn2)=O)C(C)C)cccc1S(N)(=O)=O CCC(O)C(C)C(=O)NC1(CNC(=O)CCNc2ccccn2)CCC1 c1(NC(C2C(O)CCN(C(C(CC=C)OC)=O)C2)=O)cnc2n1CCOC2 C(C)(C)(CC(=O)N1CCC(CCC(N2CCCCCC2)=O)C1)OC c1(C(N2C(C3CCN(C(C(C)OCC)=O)CC3)CCC2)=O)cc2n(n1)CCCO2 N1(CC(=O)NC2(NC(=O)CN3CC4CC4C3)CCSC2)CCC(CO)CC1 C12(C(N3CCC4(CC(NC(C56CC(C5)C6)=O)C4)C3)=O)CC3CC(C(=O)N1)C2C3 CC(C)CC(C(=O)NCCN1CCCC1=O)NC(c1cnn(C)c(=O)c1)=O C12(CNC(=O)C(C3CCCCC3)O)CC(CO1)N(C(c1ccnc(CO)c1)=O)C2 C#CC1CCCN(C(C2(NC(=O)Cc3nc(=N)[nH][nH]3)CCCC2)=O)CC1 c1(OC)cc(-c2cncnc2C(=O)Nc2ccc(C)nc2I)cc(C)c1 N1(C(c2cc(CSCC)on2)=O)CCC(F)(CNC(C2CCCC2C)=O)CC1 S(=O)(=O)(CCC(=O)N1CCN(C(=O)CN2CCCNC2=O)CC1C(C)(C)C)NC C(C)(CC(=O)N(C)CCN(C)C(c1cnn(C2CCCCC2)c1)=O)SC CC(C)CC(C)(O)C(=O)NC1CCC(C(=O)NC2CC3CCC(C2)S3)C1 c1(OC)ccc2nc(C(c3nnnn3C3COC3)NCC(F)C3CCC3)sc2c1 C=CC1(CC(=O)NCCCNC(=O)C=Cc2ccc(CC)cc2)CCOCC1 C1(C(=O)NCC(CC)NC(c2c(Br)noc2C)=O)CC2C=CC1C2 CC(C)C(C)C(CNC(=O)CCc1cnn(C)c1)NC(C1(S(N)(=O)=O)CC1)=O C(=O)(C#CC(C)(C)C)N(C1CN(C(=O)C(C)(C)n2cccn2)C1)C.C1(N)CCC1O C1(C)(C(=O)NCC2C(NC(C(C)OC3CCOC3)=O)C2)CCN(C)CC1 C(=O)(C(C(F)(F)F)=Cc1ccccc1)N1CCCC(NC(C2CC2F)=O)CC1 Cc1cc(C(=O)NC2CCCC2CNC(c2n[nH]cc2Cl)=O)cc(C)c1C C1(CNC(CCC=C(C)C)=O)CCC(NC(=O)CCN2CCCC2)CC1 C(=O)(C(C)(C)C(N)=O)NC1C(NC(c2c(C(=O)OC)coc2)=O)CCC1 c1(C(N(C)CC2CCCS2(=O)=O)=O)ccc(-c2cc[nH]c(=N)c2)cc1 c1(C(=O)NC2CC(NC(c3c(Cl)cc(C)s3)=O)C2)cc2ccc(Br)nc2[nH]1 CC(CCN=c1nc(C(C)(C)C)[nH]s1)NC(C1CCCCN1C)=O N1(C(C(C)=CCC)=O)CC(N(C(=O)CSC(F)(F)F)CC)CC(C)(C)C1 c1(CCNCC(C)CNC(=O)OC(C)(C)C)cncc(Br)c1 C1(C(=O)NC2CN(C(c3cc(Cl)no3)=O)C2)C2CS(=O)(=O)CC12 c1(C(CC(=O)OC)NC(=O)C(O)C(C)OC)cc(OC)cc(OC)c1 c1(C(=O)NCC2CCC(NC(C(C)C(F)(F)F)=O)C2)nnc2n1CCCCC2 N1(C(CCCC(=O)N(C)C)=O)CCC2CCN(C(c3csc(CO)n3)=O)CC2C1 C1(OC)CCN(C(=O)C(CC(F)F)NC(=O)Cc2ncccc2F)CC1F n1(CC(=O)N(C2CCN(C(=O)Cn3cnnc3O)CC2)C)nc(C(F)F)cc1C C(C(=O)N1C(C(=O)NCc2cnc[nH]2)CCC12CC2)(C(C)(C)C)N(C)C C1(NC(CCNC(=O)OC)=O)CCCCC1NC(c1cnn(CC2CC2)c1)=O N1(C(C(CCC)N(C)C)=O)CC(C)(C)CCC1CNC(=O)CCCS(C)(=O)=O N1(C(C(c2ccc(C)s2)C)=O)CCC2CN(C(C3CCCCO3)=O)CC2C1 c1(C2C(C(=O)OC)C2)ccc2nc(C(N3CC(C)(O)C3)=O)cn2c1 Cc1o[nH]c(=NC(=O)C2CCCn3c(C(=O)NC(C)(C)C)nnc32)c1Br c1(CCC)ccc(N)c(C(=O)NC2(CNC(=O)CCS(C)(=O)=O)CCCCC2)c1 N1(C(C(C)(C)Br)=O)CCC2C(CCN2C(c2ccc3ncnn3c2)=O)C1 N1(C(CCC#C)=O)CCC(n2cc(CC)nn2)CC1.c1(C=O)ccccc1 C(=O)(CN=c1cc(C)[nH]c(=NCC2CC2)[nH]1)NCCC S(=O)(=O)(c1ccc2c(c1)OCCO2)N1CC(C(N2CC(O)CC2CO)=O)NCC1 CC1(C)C(C)(C(N2CCC(CCNC(=O)CC3CCS(=O)(=O)CC3)C2)=O)C1(C)C C1(C(CC)O)CCCN1C(=O)C(c1cn(C)nn1)NC(=O)CN1CC(C)(C)C1 CCC(C(N)=O)NC(=O)C(Cc1ccoc1)NC(=O)Cc1cccn1C C(=O)(C(C)(C1CCC1)NC(C1CC1C(C)(F)F)=O)NC(C)C(C)F N1(C(c2cnc(Cl)s2)C(=O)NC(CC)C)CCOC(C(F)(F)F)C1(C)C C1(C)(CNC(c2cc(OCC)n[nH]2)=O)CCN(c2nnc(C(F)(F)F)s2)C1 N1(C(C2N(C(C)C)C(=O)CC2)=O)Cc2nccn2CC(NC(C2(O)COC2)=O)C1 c1(CCCC)nc(C)c(CC(=O)NC2CC(CNC(=O)C#CC(C)C)C2)s1 CCCCCCC(C)NC(=O)C(C(C)OC)NC(c1cc(C)c(C)o1)=O CCC(CC(=O)NC(C1CCN(C(=O)C=NOC)CC1)(C)C)C(=O)OC(C)(C)C Cc1ccc(C(F)C(=O)NCC2(C)CCCN2C(=O)CO)cc1 C(=O)(C(C)S(=O)c1ccccc1)N1CC2(CCC(NC(C3(OC)CCC3)=O)C2)C1 Cc1ccc(-c2cn(CC3CC3)nn2)cc1NC(=O)C(C)Cc1cnn(C)c1 c1(C(=O)NCC2(C)CCN(C(c3ncccc3F)=O)C2)ccn2ccnc2c1 N(C(=NCCCF)NCc1ccc(F)c(O)c1)C1CCCC(C(N(C)C)=O)C1 C(=O)(C#CC1CCCOC1)N1CCCC(N(C(c2ncc(OC)cn2)=O)C)CC1 C1(CC)CCN(C(=O)CN(C)C)C1C(=O)N(C(C)CN(C)C(=O)NC)C N1(C(c2cc(C)c(C)o2)=O)CCC2(CC1)CC2(CO)CNC(=O)C(C)(O)C(C)C C=CCC(C(=O)NCC=CCC(N1CCC(O)(C(N)=O)CC1)=O)C(C)C CC1(C(N2CCC(C(C)(O)CNC(=O)CC3CSCCS3)CC2)=O)CC(C#N)C1 C=CCCCC(C(=O)NCCC(F)(F)F)NC(=O)CC1CC2(CCC2)C1 C(C)(C)(CC(=O)NOCC(O)C(C)(C)C)n1cc(NC(CS(CC)(=O)=O)=O)nn1 c1(C(=O)OC)c(C)nc2c(NC(=O)C=CCF)cccn12 C1(NC(c2n(CC)nc(C3CC3)c2)=O)CCN(C(c2cncnc2)=O)CC1CO C(=O)(C1=NNC(=O)CC1)N1CCC(=CCNC(c2nccc3c[nH]nc23)=O)CC1 c1(OC)ccc2[nH]c(=NCC=CCNC(=O)C(C)(C)OC)sc2c1 Cc1ccc(C(=O)O)cc1CN(CC(C)NC(c1coc(C(C)C)n1)=O)C c1(C(N(C(C)CNC(c2cscc2Br)=O)CC)=O)cccc(F)c1O c1(CC(=O)NCCC(C)NC(=O)CN2CCOCC2)csc(C2CCOCC2)n1 C12(NC(C3C4CCC(F)(F)C34)=O)CC3CCC(C1C2)N3C(C1CCOCC1)=O c1(N2CCC(N(N3C(C)(C=O)CCC3)C(C)=O)CC2)ncnc(C)c1F.CO c1(C(=O)NC2(CNC(c3cnc[nH]3)=O)CCCC2)cnc2c(c1)CCS(=O)(=O)C2 CC1CC2CN(C(=O)CONC(=O)C=Cc3cnn(C)c3)CC12 O=C(C(CC=CCl)c1ccccc1)N1CCC(NC(C2(O)CCC2)=O)C1 c1(C(N2CCC(C(C)NC(c3csnc3Cl)=O)C2)=O)c(Cl)n[nH]c1C1CC1 C1(N(C(CCC(c2ccc(SC)cc2)=O)=O)C)CCCN(C(C2CC2F)=O)CC1 N1(c2n(CC(C)CO)c(C3CC3C(N)=O)nn2)CCNC(=O)CC1 c1(SCC(=O)NCC(CNC(=O)CCC2CC2)OC)cc(C)c2ccccc2n1 N1(C(Cc2ccn(CC)n2)=O)CC(F)CC1CC(=O)N(CC(O)COC)C N1(C(C(C)OCC)=O)CCC(CC(C)NC(c2ccnc(CC)c2)=O)CC1 c1(NC(C(=O)O)CC(NC2CCn3nnc(Br)c32)=O)ccc2c(Br)cncc2c1 CC1(C#N)CCN(C(=O)C(CC2CCCC2)NC(=O)CC2CCC(=O)C2)C1 Cc1ccc2c(C(=O)NCC(CC(C)C)NC(C3COCC3(C)C)=O)coc2c1 N1(C(CCC=C)=O)CCN(C(C2CCSC2)=O)CC1c1ccc(OC)cc1 C1(CNC(c2occc2Cl)=O)CC(F)(F)CN1C(=O)C(C1CCCCC1)O c1(C(N(CCNC(C(C)Cc2cccc(F)c2)=O)C)=O)ccc(O)nc1Cl CCC(CC)C(F)C(=O)NCC1C=CC(NC(c2c(F)cc(Cl)cc2F)=O)C1 C1(NC(c2cn(C(C)C)nn2)=O)CCCC(N(C)C(C2(CCF)CC2)=O)C1 N1(CC2(c3cccc(F)c3)CCC2)CC(=O)N(NCC2C(C(C)C)OCCC2)C1=O Cc1nc2ncc(C(N3CCOCC(NC(=O)CN4CCCCC4)C3)=O)cc2o1 C(=O)(CS(=O)c1ccc(Cl)cc1)NCCC1CN(C(c2ncn(C)n2)=O)C1 CCCC(CCO)N=c1cccc(S(=O)(=O)N(C)CC2(OC)CCOC2)[nH]1 C1(CCOC)CN(C(c2ccc(Cl)cc2C)=O)CCN1C(c1cnc(C)nc1)=O N1(C(=O)C=Cc2nccs2)CCOC2(C1)CN(C(c1ccc3c(c1)OCO3)=O)C2 C1(C(=O)NC(c2cnn(C)c2)C)N(C(C2C=CCS2)=O)CCC1(C)C C(N=c1[nH]c2ccc(S(=O)(=O)NCC3(F)CCC3)cc2s1)c1cc(=N)[nH]cc1 N1(C(c2cn(CCC)nc2)=O)CC2CCC(C1)N2C(=O)CC1=CCOCC1 c1(Cn2c(CC(CC)C3CC3)nc(-c3ccsc3)n2)nc2ccccc2o1 c1(C(=O)NCC(C)NC(c2cc(OCC)n[nH]2)=O)cc(O)ncc1Br N1(C(C=NOC)=O)CC(NC(C2(c3cccc(Cl)n3)CC2)=O)CC2(CC2)C1 c1(OC)coc(C(=O)NC(CNC(=O)CSc2ccccc2)C(C)C)cc1=O C(CSC1CCC(C(C)C)CC1)(CC(=O)Nn1cc(C2C3COCC23)nn1)OC CC1c2c[nH]nc2CCC1C(=O)N(C)CC1CN(C(c2cc(Cl)nc(Cl)c2)=O)C1 C1(=CC(=O)NC2C(OC)CN(C(C(CCSC)OC)=O)C2)CCCCC1(C)C c1(CNC(N(CCCN(CC)CC)C)=O)ccccc1-n1cncn1 C(=O)(CCC(F)(F)F)NC(CN(C(C(C)N1CCCC1)=O)C)(C)C C1(OC)CCC2(C(=O)NC(C(=O)NCCC3(C)CCOC3)C(C)C)CC12 C1(NC(c2ccc(Cl)s2)=O)C2CC3CN(C(C4CN5CCCN4CC5)=O)C1C3C2 C1(NC(C2CC(C)(C)C2)=O)CCN(C(c2cccnc2O)=O)CC1O CC(C(=O)N(CCCNC(=O)Nc1nccs1)CCO)c1ccco1 N1(C(Cn2ncn(C)c2=O)=O)CCCC(C2CC2NC(c2cnnc(O)c2)=O)C1 N1(C(c2ccc(C)cc2)=O)CCCC2(NC(c3ccc(C)cc3F)=O)CCCC12 Cc1cc(C(N2CCOCC2CN(C)C(C2(C(F)F)CCCC2)=O)=O)c(C)s1 CC1=CCSC1C(=O)N(CCC(=O)N(C(C)CC1CC1)C)CCO C1(NC(CCC(=O)NCC)=O)CC(C(=O)NC2CC2C(=O)NC)=CC1O C1(C(=O)NCC(C(C)C)NC(C2CN(C(C)C)C2)=O)CCOC(C)(C)C1 c1(C(N2C(C)(CC(N3C(C)CC3CO)=O)CC2)=O)ncc(F)cc1N C1(CC(=O)NCC(C)NC(C2(C(=O)NC)CC2)=O)CCCN1Cc1ccncc1 C(C(C)(O)C(C)(C)C)NC(COC1(C)CN(C(CC2CC(C)C2)=O)C1)=O CONC(=O)C(=O)N1CCCC1C(=O)NOCc1cccc(C)c1 c1(OC)ccc(NC(C2CC2NCc2ccc(N(C)C)cc2)=O)c(C)c1C Cc1nccc(C(N2CCC(CNC(c3cn(C)nn3)=O)C2)=O)n1 c1(C(=O)NC(C)CC2CN(C(c3ccc(C(C)(C)C)[nH]3)=O)C2)cc(C#N)c[nH]1 C1(C(N2C(CN(C(CC3CC(OCC)C3)=O)C)CCC2)=O)CCC(C)C(C)C1 N1(C(C2CC(NC(c3c(C)n(C)cc3)=O)C2(C)C)=O)CCn2nccc21 c1(C(=O)NC2C(NC(c3ccc(-c4ccco4)s3)=O)C2)ccc(O)cc1F c1(CC(C(=O)N2CCC(n3ccnn3)C2)NC(C2CC(C)C2)=O)cnn(C)c1O O=CN1CCCC1C(=O)NC1CCCC(NC(c2cnoc2-c2cccs2)=O)C1 Cc1nnccc1CNC(=O)CCN(C(=O)C(C)(C)C1(O)CCC1)CCCO N1(C(CC(CC)CN(C)C)=O)CCN(C(c2cnc(C(C)C)[nH]2)=O)C2(CCC2)C1 c1(C(=O)NC2CCCC2NC(c2cnc(O)o2)=O)ccc2c(c1)CCC=C2 CCCC(C)(O)C(=O)NCC1C(C)CCN1C(c1cc(C2CC2)nnc1O)=O N1(CC(=O)NC2C(CC)N(C(=O)C(C)n3cccc3)CC2)C(=O)C(=O)N(C)C1=O C1(NC(C(CSC)OC)=O)CCN(C(=O)CC2(CO)CCCC2)CC12CCC2 C1(C(=O)NCC2(OCC)CN(C(C3CC3C(N)=O)=O)C2)Cc2cc(C)ccc2O1 C1(NC(=O)Cc2ccc(Br)nc2)CC2(C1)CN(C(=O)Cc1cccc(F)c1)C2 C1(C(=O)NC(CNC(C2C(C)CCO2)=O)C2CC2)CC2(C1)CC1(CCC1)C2 CC(CC(=O)N(CCCCNC(=O)C(CN(C)C)c1ccccc1)C)C(C)(C)C Cc1cc(C#N)cc(C(=O)NC2CCCC(NC(C3CCCN(C)C3)=O)C2)n1 C(=O)(C(CC(C)C)C(N)=O)NC1C(CO)CCN(C(c2nc(CCC)oc2)=O)C1 C1(CC(N2CC(F)(CNC(C(C=CC)O)=O)C2)=O)CCCS(=O)(=O)C1 c1(C(=O)NCCCNC(CC)=O)nc(Cc2ccccn2)no1 C(=O)(C1=COc2ccccc2O1)N1CCN(C(Cc2cn(C)nn2)=O)C2C1C2 C(CCS(=O)(=O)c1cccc(C)c1)N1CCOCC1.Cc1ccc(N2CC2)cc1 N1(C(c2cc(CSCC)on2)=O)C2CCC1C(CNC(=O)Cc1csc(S)n1)C2 N1(C(C(C(C)C)F)=O)CCC(C2(NC(c3ccc4ncnn4n3)=O)CC2)C1 c1(OC)ccc(C(=O)NC(C)CCCNC(=O)C(C(C)C)OC)c(C)c1OC N1(C(CC=C)=O)CCCN(C(c2[nH]nc3ccncc23)=O)CC1C c1(CCC)ccccc1C(=O)NCCOCCCN(C)C(C1CCSC(C)C1)=O N1(C(Cn2ccc(C)n2)=O)CCCC(CC(=O)NCC(CO)N(C)C)C1 N1(C(C(c2ccc(C)s2)C)=O)CCN(C(c2c([N+](=O)[O-])cnn2C)=O)CCC1C CCC(C)(C)C(O)C(=O)N1CCCCC1CN(C)C(c1nc(Br)c[nH]1)=O c1(C(N(CC(C)NC(C2OC3CCC2CC3)=O)CC)=O)cn2ncccc2n1 C(=O)(N1CCCc2ccnn21)c1ccc(NC(c2cc(C)[nH]n2)=O)nc1 N1(C(C2N(c3ccnc(SC)n3)CC(F)(F)C2)=O)CC(C)OC(C)(C)C1 c1(C(=O)NC(C)C(CO)NC(c2ccnc(O)c2)=O)ccc2ncc(Br)n2c1 C(CC)(CCCCC)(c1n(CC)nnn1)NCCS.c1cccc(N(C)C)c1C Cc1nc(CO)ncc1NC(=O)CCC1CC(CC2CCOC2C)C1 C(c1ccc(C(N)=O)o1)=CC(=O)NC(C)CN(C(=O)C(c1ccccc1)F)CC C1(NC(c2ccc(O)cc2)=O)CC(O)CN(C(c2cccc(Cl)c2Cl)=O)C1 c1(CC)nc(C)oc1C(=O)NCCn1ccc(C(=O)NCCC(=O)NC)c1 C=CC(C)CCN=c1nc(NCc2ccc(C3CC3)cn2)c2c([nH]1)CCS2 CC1(NC(=O)Cc2cccc(OC(F)F)n2)CCN(C(=O)COC(F)(F)F)C1 c1(C(=O)NC2CCC(C(=O)NCC(=C)C)C2)ccc(OC)nc1 C1(OC)CN(C(=O)Cc2cccs2)C(C)(CNC(=O)Cc2c(C)cnn2C)C1 C1(N(C(C2C(C(C)C)(CC)C2)=O)C)CCN(C(C23CC(CO2)C3)=O)CC1 N1(C(C2(COC)CCCC2)=O)CCN(C(=O)CCNC(=O)COC)C(C(C)C)C1 c1(C(=O)NCCC(C(C)C)NC(=O)Cn2cc(C#N)cn2)nc(Cl)ccc1F N1(C(C(C)NC(=O)OC)=O)CCOCC1CC(=O)NCC(C)SC N1(C(c2c(OC)csc2)=O)CCCC(C2CN(C(c3cc(I)ccc3Cl)=O)C2)C1 N1(C(C23CC(C)(C2)C3)=O)C2CCC1CN(C(c1c[nH]nc1[N+](=O)[O-])=O)C2 Cc1ccc(C(=O)NC2(C(=O)N(C)CCC3CC3)CC(F)C2)c(O)c1 C1(C(N2C(C)CNCC2)=O)CCN(CC=CCl)C2CCCC12 C1(C(C)(C)O)(CNC(C2CC2CF)=O)CN(C(=O)C(C2CCOCC2)F)C1 Nc1ccc2nc(N3CCC(NC(C4CC5CC4C4C5C4(F)F)=O)CC3)sc2c1 C1(CCNC(=O)CSc2n[nH]c(C)n2)(OC)CN(C(=O)Cc2cnn(C)c2)C1 C12(C(=O)NCC(C)(C)NC(c3cc(C)c(C)s3)=O)CCCCN1CCC2 CCCCCC(CCCCC)CC(=O)N(CCCNC(=O)C1=CCCCO1)C c1(OC)cc(C)sc1C(=O)NC1CCN(C(C2(C(C)C)CCCO2)=O)CC1 C1(C2CCCC2)(C(=O)NCC2N(C(c3c(C)cns3)=O)CCCC2)CCNC1=O C(N=c1[nH]n(C)c2ncc(I)cc12)C1N(C(=O)OC)CC(F)C1 S(=O)(=O)(c1sccc1I)NC(C(=O)OC)C(C)(C)C.C(C[Si](C)(C)C)O c1(C(N2C(CC)CC(C)C2)=O)ccc2c(n1)CN(C(C1CCS1(=O)=O)=O)CC2 C=C1CCN(c2ccnc(N3CCOC(c4ccc(C(F)(F)F)cc4)C3)n2)CC1 N#Cc1cc2cccnc2nc1N.C(CCCO)C1CC1 C(=O)(C(C(C)C)N1CCCC1=O)NC(CCNC(COCc1nnc(C)s1)=O)C N1(C(CC=C)=O)CC2(CCC2CNC(c2cccc(CF)c2)=O)C1 c1(COC)ccccc1C(N1CCCC1CN(C)C(c1ccsc1C)=O)=O C1(COC)(NC(=O)C(C2CCCCCC2)C)CCN(C(c2cc(=O)n(C)o2)=O)C1 c1(C(c2nnnn2C)NC2(COC)CCCSC2)nccc(Cl)c1C C1(C)(NC(c2cc(CC)sn2)=O)CCCCC1C(=O)NCc1ncc(C)[nH]1 N1(C(C2CN(C(=O)NC)C2)=O)C2CCC1CN(C(C1CC(SC)C1)=O)C2 c1(CN2C(NC(=O)C(c3ccccc3)O)CC3CC32)c(Cl)cccc1B(O)O c1(C(=O)NCC2(NC(CSC)=O)CCCCC2C)ccc2c(c1)OCO2 C1(C(C(=O)N(C(CC)CC)CCO)C)CC2CCC1CC2 c1(C(=O)NCC2C(NC(CCNC(C)=O)=O)C2)ccc(F)cc1O.C1COCCO1 O=S1(=O)CCCC2(CCN2CC2CCCCCO2)C1 C(C(C)(C(N)=O)NCC12COCC(c3ccccc3)(C1)C2)OC c1(CC)cc(C)ccc1C(C)C.N12CCC(CC1)N(CC)C(=O)COC=CC2=O CCCC(C(=O)NCC12CC(NC(c3ncc(Cl)nc3Cl)=O)(CO1)C2)C(C)C N1(C(C=C(C)C)=O)CCC2(CC1)CC2C(=O)NCCn1ncccc1=O C1(C(=O)NCC(C)(CO)NC(c2cc3c(s2)CCC3)=O)COc2ccccc2C1 C(C(=O)N1CCN(CCCOCC(=O)N)CC1)(C(C)(C)C)N(C)C.C1(CC)CCCO1 N1(C(C(CCSC)O)=O)CC(C(=O)NC2CC(OC(C)C)C2)C(C2CC2)C1 c1(C(=O)NC2CN(C(c3c(Cl)ccc(Br)c3F)=O)C2)cc2ccccc2c(Cl)n1 C12(C(=O)NCC(CNC(C3CCCN(CC(C)C)C3)=O)(C)C)CCC(C)(CO1)C2 C1(OC)(OC)CC2(COC(COC(c3ccn(CC(F)(F)F)n3)=O)C2)C1 Cc1ncc(NC(C2CC(F)(F)CN2Cc2ccccn2)=O)cc1Cl c1(C(N2CCN(C3CN(C(C4(C)CC4F)=O)C3)CC2)=O)cn2c(n1)SCC2 Cn1cc(S(C)(=O)=O)c(C(=O)NC2CC2NC(=O)CCCN2CCCCC2)n1 Nc1cc(C(N2CC3CC(NC(c4csc5nnsc45)=O)C2C3)=O)cc(O)c1Cl C1(NC(c2ccc(C)nc2O)=O)CC2(CCN(C(c3cnc(O)cc3C)=O)C2)C1 C1(c2nc(C)on2)CCN(C(c2csc(C(C)C)n2)C(=O)NCCCSC)CC1 N1(C(CCCC(C)C)=O)CCCC12CCCN(C(=O)CCCc1ccncc1)C2 CC1(C)COC(CC(N2CC(O)(CNC(C3CC4CCCCC34)=O)C2)=O)CO1 CCC(C)C(=O)N1CC(CC(C)NC(c2nncn2C(C)C)=O)C1 c1(C(=O)NCC(C2CCC2)NC(C(C)OCC(C)C)=O)ccc(=O)n2c1CCC2 CCCCCCCCC(F)C(=O)OCC1CCCC1.C1(=O)C(C)NC(=O)OCCN1 CCC(C)(C)CC(=O)NC(C)(C)C(=O)NCCNC(C1CCC1)=O Cc1nc(CCNC(=O)C(F)CC2CN(C(C3(OC(C)C)CCC3)=O)C2)c(C)o1 C(=O)(C(CC(C)C)C(N)=O)NCC(=O)NC(c1nccn1C)CC C1(C(N2C(C(N(CCCc3ccccc3)C)=O)COCC2)=O)CCC2(CC1)CC2 C(c1ccccc1)=CC(=O)NCC(c1ccccc1)NC(=O)C(O)C1CC1 c1(CC(=O)NCCOCCC(=O)NCC(O)C(F)(F)F)ccccc1F c1(C(=O)NCC2N(C(c3cc(CC)cc(C)c3)=O)CC2)cc(C)c(F)cc1N C1(NC(COC(CC)C)=O)CCN(C(c2cccc(SC)c2)=O)C1(C)C c1(OC(C)C)ncccc1C(N1CC=CC1CNC(=O)CN(C)CCO)=O N1(C(C(CC)C)=O)CCC(O)(c2cn(C(c3ccc(Cl)cc3)C3CC3)nn2)CC1 C12(C(N3CCC(CC=C)(NC(=O)CC4CCCCN4C)C3)=O)CCC(F)(CC1)C2 c1(C(N2CCCC(CNC(COCCCCC)=O)C2)=O)ccn2ccccc12 C(=O)(C1=C(F)CN(C(=O)C(C)CN(C)C)CC1)NCc1cncc(C)c1 C1(CNC(=O)CCN2CCCCCC2)CCCCN(C(C2CCCS2(=O)=O)=O)C1 C1(C#N)(C(=O)NC(CC)CN(C(=O)CCC(C)(C)OC)C)CCS(=O)(=O)CC1 C1(NC(C=CCOC)=O)CC2(C1)CC(NC(c1cc(C(C)C)oc1C)=O)C2 c1(C(C)(C)C)cc(C(N2CCC(NC(C3(O)CCOC3)=O)C2)=O)cs1 N1(C(c2c(C)cccc2)=O)CC2CN(C(=O)Cc3ccccc3Cl)CC12 c1(Cn2c(N3CCC(CN4C(=O)CCC4)CC3)nnn2)nc2cccc(F)c2[nH]1 N1(C(c2c(C)nc[nH]2)=O)CCC(CNC(c2ccc(=O)n(O)c2)=O)C1(C)C CC(C)(C)CCCCC(=O)NC1(C)CCN(C(=O)CC2CCCCC2O)C1 c1(C(=O)NCCN(CCCN(C)C)C)ccc2c(c1)C(C)(C)C(=O)N2C c1(NC(N(C)CC2(F)CCC2)=O)cccc([Si](C)(C)C)c1 N1(C(Cn2ncc(C#C)c2)=O)CCC(N=c2cc[nH]cc2C#N)CC1 C(CC(C)CC)(C(=O)N1CC=CCC1)NC(C(C)NC(CC)=O)=O Fc1cc2nc(NC3CCN(C4CCCCC4)CC3)sc2cc1F N1(C(C2C(C)OCC2)=O)CCC2(CC1)CC(Nc1ncnc(C(C)(C)C)n1)CO2 c1(OC)cc(CC(N2CCN(c3nc(C)cc(C)n3)CC2)=O)cc(Cl)n1 c1(NC(C2CCCC2CNC(C23CCC(C2)C3)=O)=O)ccccc1CO n1(C(C)C)ccc(C(N2CCC(CNC(c3cnn(C4CC4(F)F)c3)=O)C2)=O)n1 N1(C(C2N(C(C3CCN(C)C3)=O)CCC2)=O)CC(CO)CC12CCC2 Cc1cc(O)ccc1NC(C1CC=CCN1C(C1CCCS1)=O)=O N1(CCNC(=O)CN(S(C)(=O)=O)C)CCCN(NC(C2C(=C)CC2)=O)CC1 N(C1CCCc2c(Br)cccc21)C(c1c(C)nc2ncnn2c1)=O C(C(=O)NCc1csnc1C)(C(C)(C)O)NC(c1ccc(OC)nn1)=O c1(NCC(C2CCC2)OCC)[nH]c(=NCC2CC(C)C2)nc2scnc12 c1(CC)cc(COC(=O)CC2CCCOCC2)ccc1F CCCC(C(=O)NCC1(C(N)=O)CN(C(c2ccnnc2S)=O)C1)C(C)C C(=O)(CC1=CCN(C)CC1)N1CCCC(N(C(c2nn(C)c(Cl)c2Cl)=O)CC)C1 CC1(C)C=CC(NC(=O)CCCCCNC(C2CC=CCC2)=O)CC1 C1(CC(=O)NC(C2(C(=O)N(C)Cc3ncccn3)CC2)C)CCCCC1O c1(C(c2n(CC(=C)C)nnn2)NCC2CCCO2)cnn(CC(C)C)c1.OC Cc1ccc(C(N2CC3(CC(CNC(=O)CSc4n[nH]c(O)n4)C3)C2)=O)c(C)c1 C#CC1(NC(C2(NC(=O)CCC(C)SC)CCCC2C)=O)CCC(C)(C)C1 C1(NC(C(C(C)C)NC(N)=O)=O)CC2CCC1CC2NC(C1CC2CC2CO1)=O O=C(CCOCCNC(c1cnsc1)=O)NCCn1cnnc1 C1(NC(C2(C)C(C)C2)=O)CCOC2(CCN(S(=O)(=O)c3cccc(Cl)c3F)CC2)C1 C1(N(C(c2c(OC)ccs2)=O)C)CCN(C(C2CCC(O)CC2)=O)CC12CC2 c1(C(=O)NCC2(O)CC(NC(C=COCC)=O)C2)ccc2c(c1)C1CCC2O1 C=CCC(C(=O)N(C1CN(C(=O)C(=O)N(C)C)CC1O)C)C(C)C N1(C(C2C3COCC23)C(=O)NCC2CCOC2)CC2CCCCC2C1 c1(OC)cc(C(=O)NCC2CCN(Cc3cccs3)CC2)ncn1 c1(OC)ccccc1C(CNC(=O)C(C)CF)NC(=O)CCc1cccnc1 c12cccc(c1)NCC(O)CN(C)C(=O)CCc1nnc-2o1.c1(CC)csnn1 c1(C(=O)NCC2(COC)CN(C(C3CCSC3)=O)C2)ccnc(C)c1C c1(OC(C)CNS(=O)(=O)CCBr)ccc(Br)cc1 C1(O)(CNC(c2c(CC)n[nH]c2)=O)CC2CCC(C1)N2C(=O)Cn1cnc(=N)[nH]1 c1(CC(=O)N(CCC)CCC)ccc2cc(OC)ccc2c1 c1(C(N2CCN(C)CC2)=O)n[nH]c2ccc(-c3cc(F)c(F)cc3O)cc12 c1(CC)ccc2[nH]c(C(=O)NCCCNC(C3C4CC4C4CC34)=O)c(C)c2c1 Cc1ccc(F)c(CNC(C(C)(C)C)c2nnnn2CCCC2CC2)n1 CS(=O)(=O)CCCCS(=O)(=O)N1CCOCC12CCOC2 c1(C(=O)NCC23N(C(C4C(C=C)C4)=O)C(CC2)CC3)coc2ccc(F)cc12 Cc1ccc(CNC(=O)C(=O)NCc2cnn(C(C)(C)C)c2)cc1C#N C1(O)(CC(=O)NCC2CC(C(=O)NC3CC(O)C3)CO2)CCCOC1 Cc1cc(F)c(Cl)cc1C(=O)NCC1CC(C)N(C(=O)OC(C)(C)C)C1 c1(N2CC3CCN(C(=O)Cn4nc(Cl)ccc4=O)C3C2)ncnc2c(Br)c[nH]c12 Cc1ccc2[nH]cc(CCC(=O)NC(C)(C)C(c3ccc(Br)cc3)=O)c2c1 c1(C(=O)NC(CNC(C2C(CC)C2)=O)C(C)(C)C)cnc2[nH]cnc2c1 c1(C(=O)NCC2(CNC(C3CC(F)(F)C3)=O)CCC2)cccc(S(=O)(=O)CF)c1 n1(CCCC)nc(C)c(C(=O)NCC(C)NC(c2nc(Cl)sc2Cl)=O)c1Cl c1(CC(=O)N(CC(C)N(C(=O)C#CC2CC2)C)C)cc(Br)c2c(c1)CCO2 C=C=CC(C)C(=O)N1CCCC(N(C(=O)Cc2ccc(O)nc2)CCF)C1 C1(F)(C(N2CC(OCCNC(CC(CC)OC)=O)C2)=O)CCS(=O)(=O)C1 C1(C(C)(C)C)CC(C(=O)NCC2C(NC(C3(F)CC=CC3)=O)C2)=NO1 C1(CC(=O)NCC2CC(C)N(C(=O)CC3(O)CCCCC3)C2)CC2(CCC2)CO1 CN1CC(NC(c2cc(CNC(C3(C)CCC(=O)C3)=O)nn2C)=O)C(=O)N1 C(=O)(C1=CCCCC1)NCCNC(CC(c1ccc(C(C)C)cc1)C)=O c1(C(N2C3(CNC(C(CC)(F)F)=O)CC(C2)C3)=O)cc(C)n(C2CCOC2)c1C CCCC(C(=O)NCC1(O)CC(CNC(c2cc(C)c(C)s2)=O)C1)OCC N1(CCC(=O)N(C2CCN(C(=O)CCCOC(C)C)C2)CC)CCCCC1 C(=O)(C1CSc2ccccc21)N1CC(CC(C)NC(CCc2scc(C)n2)=O)C1 C#Cc1ccc(C(=O)NC2CC2NC(=O)Cc2ccccc2NC(C)=O)cc1C C1(C(=O)NCC(C)NC(c2c(OC(C)C)cccc2)=O)CCCCC12CC2 C1(NC(C(C)OCCC=C)=O)C(C)CCN(C(c2ccc(C)c(N)c2)=O)C1C C1(CNC(C2ON=C(C)C2)=O)CC2CCC(C1)N2C(c1ccc2[nH]ccc2n1)=O C1(NCC2(C)N=C(C)SC2)CCCCCC1C N1(C(CCC#C)=O)CCC2(C=C(C(=O)NCCc3ccncc3C)C2)C1 C(C(C)CC(=O)NC1CC(CNC(=O)C(C)NCC(F)(F)F)C1)OC C1(C(=O)NCC2CN(C(C)C)C2)CN(C(C2CCS2(=O)=O)=O)CCO1 CC(=O)CCCC(C)C(=O)NC(CC1CC1)CC(=O)Nc1cccc(N(C)C)c1 C1(C)(NC(C(C2CN(C(=O)C(O)CCN(C)C)C2)OC)=O)CCC2(CC1)CC2 CC(C)CC(F)C(=O)NCCN(C(c1ccc(Br)cc1OC)=O)C(C)C c1(CC)ccncc1NC(=O)CCNC(=O)C(C)NC(C)=O C1(CC)CC(C(=O)NCCCOCCN(C)C(C2CC(C(=O)OC)C2)=O)C1 C=CCCCCCCNC(=O)C(C(C)(C)O)NC(=O)CNC(=O)C(C)CC N1(C(c2c(OC)ccc(C)n2)=O)CC2CC(C1)N(C(=O)Cc1cnn(C)c1C)C2 N1(C(c2ccc(CC)s2)=O)CCC2CN(C(=O)Cc3ccccc3)CCC12 N1(C(c2cccc(C(C)(C)C)c2)=O)CC2(CCC2CNC(c2cn[nH]c2)=O)C1 CC1CC(CNc2cccc(NC(C3(NC(N)=O)CCCC3)=O)c2)CCO1 N1(C(Cc2cccc(OC)c2)=O)CCN(C(=O)C2=NOC(C)C2C)CC12CCC2 C(=O)(C(C(C)C)C(C)C)NCC(C)N(C(=O)C(O)Cn1cncn1)CC CCCCCCS(=O)(=O)N1CCC(C(=O)Nc2ccc(N(C)C)cc2)CC1 C(=O)(C(C(C)(C)C)C1CCC1)NC1C(n2cc(C(CC)(C)C)nn2)CCC1 C1(C(=O)NC(CNC(CCOCCOC)=O)C(C)(C)C)COCC(=O)N1C(C)C c1(C(=O)NCC2CN(C(=O)CSC3CC3)CC2C(F)(F)F)cc2c(cc1Cl)NCC2 C(=O)(C1=CCCC1)NCC1(CN(C)C(C2CC3(C2)CC3F)=O)CC1 C1(CNC(c2cnc(C(C)C)[nH]2)=O)CCCCN1C(=O)CCc1cncs1 N1(C(c2cc(C)c(C)o2)=O)CCCCCC(NC(=O)CC2CCS(=O)(=O)C2)C1 C(=O)(CC1=CCOCC1)NC(CCCOC)C(=O)NCC(F)Br N1(C(C(C(C)C)N(C)C)=O)CCC2(CC1)CC(C)N(C(=O)C(O)C1CCC1)C2 CC(C)CCCCC(=O)NC1CN(C(C23CCCCN2CCC3)=O)CC1CO Cc1cc(N)ccc1C(=O)NC1CCCC(NC(=O)Cc2nncn2C(C)C)C1 CP(C)(=O)C1CCC(NC(=O)NCCCN(c2ccccc2)C2CC2)C1 C=C(C)C1OCCC1CNC(=O)CN(C(C1COCC1CC)=O)CC c1(C(=O)NCCCCNC(C2C(=C)C2)=O)ccc2c(c1)OC(C)(C)C2 Cc1cc(CCC(=O)NC2(C(=O)NC3CCCC3O)CCCC2)cs1 c1(OC)ccc(Br)cc1CNc1c[nH]nc1C(N1CC2CNC(=O)C2C1)=O C1(CNC(CCOCCC)=O)COCCN(C(=O)COC2CC2(F)F)C1 C1(CC(=O)NCC2(CCOC)CC2)CCN(C(c2cc(C)cc(C)c2)=O)C1(C)C CCCCC(O)C(C)C(=O)N1CCCC(NC(c2cccc(N)c2C)=O)C1 C(C(C)C(=O)NCc1ocnc1C(=O)NCCCC(=O)N(C)C)OC Cc1cc(C(=O)NCC2CC(NC(c3cscc3F)=O)CCO2)c(F)cc1Cl C#Cc1ccc(C(=O)NC(C)C(C)NC(=O)C(C2CCCCCC2)C)c(F)c1Cl N1(C(CC(COC)C)=O)CCCC12CCN(C(=O)CC1CCC(C3CC3)O1)C2 c1(C(=O)NC2CN(C(CCC#C)=O)C(C)CC2)cc([N+](=O)[O-])cnc1O C1(O)(C(=O)NCCC2CCCN(C(=O)COCC(F)(F)F)C2)CC2CCC1C2 c1(OC)cc(Cl)ccc1C(=O)N(C)CC1(NC(c2cnc(C3CC3)[nH]2)=O)CC1 C1(NC(c2cnc(OC)s2)=O)C(C)CN(C(c2ncn(C(C)C)n2)=O)CC1C N1(C(c2c(C)nns2)=O)CCC2(CNC(=O)Cc3cccc(Cl)c3)CCCCC12 C(=O)(C(C(C)CC)N(C)C)NCc1occ(C(=O)NCCSCC#C)c1 CC(C)CCC(=O)C(=O)N1CC(F)CC1C(=O)NCCN(C(C)C)C(C)C Cc1ccc(S(=O)(=O)n2c(C(=O)NCCC3CC3(Br)Br)cc3ccccc23)cc1 N1(C(CCc2cccc(OC)c2F)=O)CCCC2CCNC(=O)C12 N1(C(C)=O)CCC(C(=O)NCC2CCCN(C(c3ccncc3)=O)C2)C(F)(F)C1 c1(CC)n[nH]c(CC)c1CC(=O)C1CC1.c1(CN)cn(CC(C)NC(=O)C(N)=O)nn1 C1(C2CC2)(C(=O)NCC(C(=O)NCCCCC(C)C)CC2CCCC2)CC(=O)C1 c1(C(=O)NCC2C(NC(CC(C)C3CCCCC3)=O)C2)c[nH]c2ncccc12 N1(C(c2ccn(CCOC)n2)=O)CCOCC1CN(C(=O)CN(C)C(C)C)C C12(CNC(CCCOC(C)C)=O)CCCCC1N(C(=O)C=CS(C)(=O)=O)CC2 c1(C(=O)NCC(CC)NC(c2nocc2Cl)=O)cc(C2(C)CC2)on1 N1(C(c2ccc(CC)s2)=O)CCC2C(C1)NC(=O)CN2C(=O)CC(C)OC N1(C(C(C(C)C)NC=O)=O)CC2(CC(NC(c3ccc(Br)c(N)c3)=O)C2)C1 C1(CNC(C(C)OCC#C)=O)C2CCC(C2)N1C(=O)CC=CC C=C(C)C(C)(C)C(=O)N1CC(O)(C(C)NC(c2cc(C)n(CC(F)(F)F)n2)=O)C1 c1(C(N(C2CN(C(CC3CCCC(C)C3)=O)C2)C)=O)cnc2c(n1)CCCC2 Cc1cc2ccc1OCS2.c1(C)nncn1C1CC1 CC1CN2CCCC2CN1C(c1nc(Cl)ccc1Br)C(=O)NCc1cccs1 Cc1ccc(C=CC(N2CCCC3(CNC(=O)CCF)CC23)=O)cc1 N1(C(C)=O)CCN(C(c2ccnc(C(C)(F)F)c2)=O)C2CCCCC2C1 N1(C(CCCC(CC)NC(=O)C(CC)SC)=O)CCc2cccc(O)c21 C1(CNC(CC=C=C)=O)CC2CCC1N2C(c1cnn(Cc2ccccc2)n1)=O N1(C(CC(C)OC)=O)CC(C2CC2)(C(=O)NCC(O)(C2CC2)C2CC2)C1 c1(C(=O)Nc2c(CC)n(-c3cccc(C(F)(F)F)c3)nc2)[nH]nc([N+](=O)[O-])c1Cl c1(C(=O)NC2CC(CNC(CCc3n(C)ccn3)=O)C2)cccc(C(C)(F)F)c1 c1(CC(c2ccccc2)NC(=O)NCCc2ncc(C)cn2)ccc(Br)cc1F CC1(C)CN(CCC(=O)N2CC(NC(=O)C=C(Cl)Cl)C2)CCS1 c1(C(=O)OCc2cncc(CC)c2)cnc2nc(C)ccc2c1O C1(CNC(C(CC)(F)F)=O)CC12CCN(C(c1cc3ncccc3o1)=O)CC2 C1(COC)(CNC(c2occc2CO)=O)CCN(C(c2ccccc2O)=O)CC1 c1(CC(=O)NC2(CNC(CC(n3ccc(C)n3)C)=O)CCCC2)ccc(O)cc1 C1(C(N(CCCN(C)C(C2CCCC23CC3)=O)C)=O)CC2CC1C1CC21 C1(C2CCCN(C(=O)C3CC3)C2)(NC(C(c2ccc(C)cc2)(F)F)=O)CC1 N1(C(C2=NNC(=O)CC2)=O)CCc2nc(-c3cccc(OCCO)c3F)sc2C1 c1(SC)ccc(S(=O)(=O)NCCn2cc(-c3ccc4scnc4c3)nn2)s1 n1(CC(=O)NC(CN(C)C(C2COC(=O)N2)=O)(C)C)cnc([N+](=O)[O-])n1 C1(C(N2C3CC(NC(=O)CN4CCSCC4)(C3)C2)=O)CC2C=CC1C21CC1 C1(C(=O)NC(CNC(C(CCN(C)C)N(C)C)=O)CO)CC12CCCCC2 CC(CC(=O)NC(CC1CCC(=O)C1)CO)C1CC1 c1(NC(C2C(NC(C(CC)C)=O)C2)=O)cnc(Br)nc1 C1(O)(C(C)NC(COCC=C)=O)CCN(C(=O)Cc2ccccn2)C1 C(=O)(C#CC(C)(C)C)NCCCCc1cn(CCC(=O)OC)nn1 N1(C(C(C2CC2)OC)=O)CCN(C(=O)CNC(c2ncoc2C(F)(F)F)=O)CC1 C1(NC(c2ncc(C)nc2)=O)CN(C(=O)CCCC2CCCO2)CC1C1CC1 c1(C(C)C)nc(CC(=O)NC2CCC2CNC(=O)CC2(C)OCCO2)cs1 C1(NC(=O)CCc2ncc(F)cn2)CN(C(c2sccc2CO)=O)CC1F N1(C(c2ccc(F)cc2F)C)CCOC2(CCN(C(=O)CN=S(C)(C)=O)C2)C1 C(C(C)(O)C(=O)NCC(C)CNC(c1ccc(SC(F)F)cc1)=O)OC c1(NCC2N(C(C3(C)CCC3)=O)CCCC2)ncnc2c(Br)csc12 C1(O)(CCNC(C2(CC(C)C)CCC2)=O)CCN(C(C2CCC(=O)N2C)=O)C1 S(=O)(=O)(CCC(=O)NC1CCN(C(=O)C(N2CCOCC2)C)C1C)NC CONC(=O)C(=O)N1CCC(c2ccccc2)(NC(=O)C(C)N2CCC2)C1 Cc1nccnc1C(N1CCC(N(C(=O)C2=CCC2)Cc2ccccn2)C1)=O c1(C(N(C2CCN(C(C(C(C)C)SCC)=O)CC2)C)=O)ccnc(Cl)c1O C1(C(=O)NCCOC(C)C)CN(C(C2CCCSC2)=O)C2(CCC2)C1 c1(SC(C)C(=O)NCC2(F)CC(C(=O)O)C2)nnnn1C1CCCC1 n1(CC)ncc(C(N2CC(NC(c3cc(C4CCC4)nn3C)=O)C(C)C2)=O)c1C c1(-c2cnc(C(=O)Nc3cc(OC)c(F)cc3Br)nc2)ccc2cnn(C)c2c1 C12(CC(=O)NC(COC)(C)C(=O)OC)CCC(CC1)CN2C(=O)OC(C)(C)C N1(C(=O)CN2CCCC3(CC3)S2(=O)=O)CCCCC2(CCOCC2)C1 C=CC1CN(C(=O)C(Br)=C(C)C)CC1NC(c1ccc(OC(C)C)cn1)=O C(=O)(C#CC1CCOC1)NC(c1ccc(C)cc1)CNC(=O)Cc1nc[nH]n1 N1(c2cc(C)nc(Cl)n2)CCCC12CCN(C(C1CCCCS1)=O)C2 N1(C(c2c(CC)ccc(F)c2)=O)CCC(N=c2[nH][nH]c(=N)[nH]2)CC1 c1(CC)ccccc1C(=O)N(CCCC(=O)NCc1ccc(C(N)=O)o1)C C1(C(N2CCC(N(C(=O)CCOC3CCCOC3)CC)C2)=O)CC(C)(C)CCO1 N1(C(C(c2c(C)nn(C)c2C)C)=O)CC2CN(C(=O)C3=NNC(=O)C3)CC2C1 C1(C(=O)NC2C(CN(C)C)CCC2)C2CCN(C(C3(F)CCCC3)=O)CC12 Cc1ccc2[nH]cc(C(=O)NC3CCN(C(c4cc[n+]([O-])cc4)=O)CC3C)c2c1 CC(CC(=O)N1CC(NC(=O)C2=NOCC2)C2(CC2)C1)P(C)(C)=O c1(CC(=O)NC(CSC)C(C)C)c(C)cc(C)cc1C.C1(C)(C)C=CC(=O)N1 N1(C(c2c(CC)cco2)=O)CCC(NC(c2c(C)cc[nH]c2=N)=O)C(F)C1 Cc1cc(CCCC(=O)NC(C2(O)CN(C(=O)C(n3cc(Cl)cn3)C)C2)C)on1 C1(CNC(CCC2(C)CC2)=O)CCCCN1C(c1ncnn1C1CCCCC1)=O N1(C(C(C)N(C)Cc2ccccc2)=O)CC2CCCC1(NC(c1ccsc1)=O)C2 c1(NC(C2CC(CC)C2)=O)cccc(Cc2ccc(Cl)cc2)c1 c1(C(N2CC3C(NC(C(C)C(C)(C)C)=O)C3C2)=O)cc2cc(F)ccc2[nH]1 O(NC(=O)C(Cc1ccoc1)NC(=O)C1=NOC(C)C1)CC(=C)C CCC(CC(=O)NC1CC2C(NC(C3CSCN3C(C)=O)=O)C2C1)C1CC1 C12(C(=O)OC)CC1CN(C(c1csc(Cl)c1)C(=O)NC1CCCC1)C2 CN1CCC(C(N2CCCC2CNC(c2c[nH]c(Br)c2)=O)=O)CC1=O N#CC1CCCC(C(N2CC(C3CC3)(C(N3CCN(C4CC4)CC3)=O)C2)=O)C1 C(=O)(CCCC(C)=O)N1CCCC(N(C(C2CC3(CSC3)C2)=O)CC)C1 C1(CCC)(NC(c2cnc(OC)nc2)=O)CCN(C(c2cc[nH]c(=N)n2)=O)CC1 C=CCC(Cc1ccccc1)C(=O)N1CC(C)C(N)C1.c1ncno1 CC(C)C(C(=O)NC1CC(C)(CO)C1)NC(=O)C(O)CNC(N)=O NC(=O)CC(N)C(=O)NC12CC1C2.c1ccc(F)cc1.C[Si](C)(C)C C(c1ncccc1C)=CC(N1CC(CCNC(=O)CC2CCCCO2)(OC)C1)=O C1(NC(C(C)(C)OCC)=O)CC2CC1N(C(c1ccc(N(C)C)cn1)=O)C2 Cc1cc(F)c(N)cc1C(N1CC(OCCNC(C2CC3CCC2C3)=O)C1)=O c1(C(=O)NC2CCCC(NC(c3ccc(F)o3)=O)C2)ccc2n[nH]cc2c1 CC(CC(=O)N1CCC(NC(c2cc(C3CC3)[nH]n2)=O)C1)c1ccco1 CC1=NOC(C(=O)NC(Cn2ccnn2)C(=O)N(C)Cc2nnc(O)o2)C1 N1(C(C2(NC(C(C)NC(C)=O)=O)CC2)=O)CCC2(C=CCO2)CC1 c1(-c2onc(C)n2)ccc(C)c(C(N2CCCC(O)(C(F)F)C2)=O)c1 Cc1ccc(C(=O)C(=O)NC2CC(NC(c3csc(Cl)n3)=O)C2)cc1 C1(S(=O)(=O)c2ccccc2)(C(=O)OCc2n(C)ncc2Br)CCOCC1 c1(C(C(=O)N(CCNC(C(C(C)O)N(C)C)=O)C)(F)F)ccc(=O)n(C)c1 c1(C(N2CCC(NC(C(C)SC)=O)C(O)C2)=O)ncc(P(C)(C)=O)cn1 N1(C(C2(CC=C)CC2)=O)CC2(CC(NC(=O)C(C)(C)Cc3ccccc3)CO2)C1 N1(CCC(=O)OC)C(=O)CCC1CC1CCN(C(C)(C)C)C1 C(=O)(C(F)(F)C(F)(F)F)NCC(C)N(C(C(C1CCOCC1)OCC)=O)C c1(C(=O)OC)cc(C(=O)NCC(C)CNC(=O)CC2C=NN(C)C2=O)c(C)s1 C(=O)(C(C)(CO)NC(c1ccc(O)nc1)=O)NCC(C)OC c1(C(=O)NCC2CCN(C(=O)Cc3ccc(F)c(F)c3)C2)cnn2c1OCCC2 N1(CC)CCN(CC(N2CCN(C(=O)C3=CCCSC3)CC2CO)=O)C(=O)C1=O Cc1ccc(C(=O)NC2CCCC2NC(C2CCCN2C)=O)c(F)c1F c1(C(=O)OCC=[SH]C(C)C)ccc(C(F)F)nc1O CC(C)(Cc1noc(C2(NC(=O)OC(C)(C)C)CC2)n1)CS(C)(=O)=O n1(CC)nc(C)c(CC(=O)NC2CC(F)(CNC(=O)Cc3ccncn3)C2)c1C C1(NC(C2C(C(C)O)C2)=O)CC1C1CCCN(C(c2cncc(N)n2)=O)C1 N1(C(Cc2cn(C(C)(C)C)nc2)=O)CC2CCN(C(C34CC(CO)(C3)C4)=O)C2C1 N1(C(CC2CN(C)C2)=O)CC(NC(=O)CNS(N)(=O)=O)C(C2CC2)C1 O(N=C1CCCCCC1)OC(=O)CC(c1ccc(Cl)cc1)O.C12CC(C1)C(=O)N2 c1(C(N2CC(CNC(CC(C)(C)C)=O)C3C2C3)=O)ncn2cc(Cl)ccc12 CC1(C(N2CCC(CO)(CNC(c3ccon3)=O)CC2)=O)CCCS1(=O)=O C1(C(=O)NCc2cc(C(N3CC(OCCCCC)C3)=O)no2)CC2C(C1)C2(F)F c1(N2CCCCC(C)C2)nc(=NCCC2CCCOC2)[nH]c2c1CCCCCC2 c1(C(=O)NS(C(CC)c2ccccc2)(=O)=O)cc(F)cc(F)c1 C(=O)(C1CCc2nccn21)N1CCN(C(C(CC)CC)=O)CC1CO Cc1conc1C(=O)N(CCCNC(C1CCC1)=O)CCO S(=O)(=O)(c1c[nH]ccc1=NCc1nc(C2CCCOC2)cs1)NCC1C(C)(C)C1 C(C(C(=O)N1CC2CC(N(C(=O)C(C)CC(C)(C)C)C)C1C2)C(F)(F)F)OC Cc1[nH]nc(C(=O)NC2CCCC(CNC(c3cnn(C4CCC4)c3)=O)C2)c1F C1(CNC(C2C(OCC)C2C)=O)Cc2ccccc2CN1C(C1C=CCC1)=O c1(NC2(C)CC(NC(c3c(C)noc3C)=O)C2)ncc([N+](=O)[O-])c(=N)[nH]1 C1(CNC(C2(CCOC)CC2)=O)CN(C(=O)CC2=CCCC2)CCC1(F)F c1(CNC(=O)NCC(C)CN2CCCC2)nc2c(s1)CC(C)CC2 CCC(C)(F)C(=O)NC1CCN(C(c2cn(C3CCCC3)nn2)=O)C1 C1(C(=O)NC(COCC)C(=O)N(C)CCOC2CC2)CCC(CO)CC1 N1(C(c2cn(CC)nc2)=O)CC(CNC(=O)CCC#N)CC1C N1(C(CNC(=O)NC)=O)CC2CCCC(NC(=O)C(N3CCSCC3)C)C2C1 C(=O)(C1CCCc2n[nH]cc21)N1CCC(NC(CC(CCOC)(C)C)=O)C12CC2 N1(C(C(C)CC#N)=O)CC2(CCC2)CC1C(=O)N(C(C)CC1CC1)C c1(CC)nc[nH]c(=NCC2CCN(C(c3cnc4c(c3)CCOC4)=O)CC2)c1F CC1(C)C(C(=O)NCCn2ncnn2)CCN1C(=O)Cc1ccsn1 c1(C(N2C(C)CC(CNC(C3CCC(=O)N(C)C3)=O)C2)=O)c(Cl)oc2ccccc12 O(C1CCOc2c(Br)cccc21)CC12C(C)(C)C(CC1)CC2 CC1NC(=O)CCC1NC(=O)NCC(c1ccccc1Cl)=O c1(C(N2CC(CNC(C3C(c4onc(C)n4)C3(C)C)=O)C2)=O)cnn(C)c1C N1(C(C(=O)NCCC2CCN(C(CC3CC(CC)C3)=O)C2)=O)CCN(C)CC1 N1(C(c2cn(C)nc2Cl)=O)CC2CC(NC(C3(F)CCCCC3)=O)CC2C1 C1(C(=O)NC2CN(C(c3cccnn3)=O)CC23CC3)CCC2CCC(=O)N2C1 c1(C(N2CCC(N(C(C(CC=C)(C)C)=O)CCC)C2)=O)cc(C)c(OC)c(Cl)c1 c1(C(N2CCC(C(N(C)Cc3cn[nH]c3)=O)C2)=O)ccc2cccnn12 c1(C(N2CC(O)(C(C)NC(C(C=CC)O)=O)C2)=O)cn(C)cc1C c1(C(=O)NC2CN(C(c3cc(CCC)on3)=O)C(C)C2)ccc(Cl)c(Cl)c1O N1(C(CC(CN(C)C)O)=O)CC2CCC(C1)N2C(C1CCCC(=O)N1)=O O=C(C1SCCc2ccccc21)NC1(CO)CC2CCC1CC2 C(=O)(CCN=c1[nH]ccs1)NC1CCC(CNC(C(c2cccnc2)OC)=O)C1 C1(C(C)NC(=O)CCc2ccc(SC)o2)CCC(C(N2CC(O)(C3CCCO3)C2)=O)O1 C12(OC)CCC(C(N3CCOCC(CNC(=O)C(C)C(C)O)C3)=O)(CC1)C2 C1(NC(CC2(COC)CC2)=O)CCCC(NC(c2ccc(C)cc2F)=O)CC1 C(=O)(C1=CNC2=NCCCN12)NCC(C)N(C(CCn1nc(C)c(C)c1C)=O)C Cc1c(C#N)c(-c2ccccc2)n(CCc2csc(C3CC3)n2)c1C C1(NC(c2ccn(CC)n2)=O)CCN(C(c2cn(C)nc2SC)=O)CC1CO N1(C(c2cc(C)ncc2)=O)C2CCC1C(NC(C1CC13CCC3)=O)C2 C1(C(=O)NC2CCN(C(C=CC(C)(C)C)=O)CC2O)CCCC(C)(C)CC1 Cc1cccc(C(N2CC(O)CC2CNC(=O)CSCCC(C)C)=O)n1 c1(NCC(CC)=CCC)c(Cl)cccc1Br.C12CN(CCO1)C(=O)COC2=O C1(NC(C(CCC)F)=O)(CNC(C2CCC(=O)N(C)C2)=O)CCCCC1C c1(C(=O)NC2(C3CN(C(C(CCCC)O)=O)C3)CC2)coc(S(=O)(=O)N(C)C)c1 Cc1onc(C2CC2)c1C(=O)NC(CC1CCN(C(C2(CCF)CC2)=O)CC1)C C=C(C)CCCC(=O)N1CCN(C(=O)C=CC2CCCC2)C2CC12 Fc1cnccc1N1CCCC(NCc2coc(-c3ccccc3)n2)C1 C(CCCC(=O)N1CC(NC(=O)CC2CC(C)(C)C2)C(CC2CC2)C1)N(C)C c1(NCCC(=O)N(C2CCN(C(c3ccc(Cl)o3)=O)C2)CC)ccccn1 Cc1ccc2c(C(N3CC4CCC3C(NC(C3CCO3)=O)C4)=O)c[nH]c2c1 c1(C(=O)NCCN(C(C2C(C)CCOC2)=O)C2CC2)cc2ncccc2o1 C12(NC(C(CC)OCC)=O)CCCC1CN(C(c1ncc3ccccn13)=O)C2 c1(C(=O)NC(C2CCN(C(c3n[nH]c(C)c3Br)=O)C2)C)cc(F)ccc1N N1(CC(=O)CCC2CCCC2)CCc2nnc(Br)n2CC1 N1(C(C(C)OCC)=O)CCC2(CC2NC(=O)Cc2cccc(C)c2)C1 C1(C(=O)NC2CCC(NC(=O)Cn3nccn3)C2)CC2(CCCCC2)C1 C1(NC(c2ccc(N)c(Cl)c2O)=O)CC2(CCCCN2C(c2ccncn2)=O)C1 c1(NC(=O)CC23CCCC2C3)ccnc(Cl)c1 C1(C)(C(N2C(C(N3CCN(CCC)CC3)=O)CC(=O)C2)=O)CC2C=CC1C2 c1(CC(=O)NC(C2CCN(C(c3cccc[n+]3[O-])=O)C2)(C)C)cc(O)nnc1O Cc1cc(NC(C)CCN2CCOCC2)c2ccc(C)c(Cl)c2n1 c1(C(c2nnnn2Cc2nnn(C)n2)NCCCOCC=C)ncccc1Cl N1(C(c2ccn(C)n2)=O)CCCC2CN(C(=O)CCc3cc[nH]n3)CCCC12 N(C(=NCCN1CCOCC1C)NCC1CC1)Cc1c(CC)c[nH]n1 c1(C(=O)NC2(CNC(CCCC(=C)C)=O)CCOCC2)ccc2c(c1)CN(C)C2 N1(C(C=C(C)Cl)=O)CC(F)(F)CC1CCNC(=O)CCN1CCN(C(C)C)CC1 c1(NC(C(Cc2cn[nH]c2)NC(c2c(CC)[nH]cc2)=O)=O)cc(C)c(C)cc1C c1(OCC)nc(C(=O)NC(C)CN(C(=O)C(C)n2ccnc2)CC)ns1 C(CCN(C(=O)CCc1cnoc1)C)(C(C)C)NC(CCOCC)=O Cc1ncc2n1CC(C(N1CC3C(CNC(c4cnsn4)=O)C3C1)=O)CC2 c1(CC(N2CCC(NC(C=CC(CC)C)=O)C2)=O)c[nH]c2c(C)cccc12 c1(CNC(COCCOC)=O)cc[nH]c1C(=O)N(C1CCN(C(C)C)C1)C c1(C(N2CC(OCCNC(CC)=O)C2)=O)nccc(C)n1 CCCCC(C)CCC(=O)NC(C)CC1CN(C(=O)C(OC)OC)C1 Cc1nc2ccnn2c(C)c1C(=O)NCCCCCCNC(=O)C(C)C(F)(F)F Cc1cc(C)c(C(=O)NCC2CCN2C(=O)CC2CCCN(C)C2)s1 C1(NC(C(=O)NC(COCC)C)=O)CC(C)CCC1C(C)C c1(C(N(c2ccccc2Br)C(C)C)=O)cc2c([nH]1)CCCC2=O c1(COC2CC(NC3(c4n(CC=C)nnn4)COC3)CC2OC)nn(C)cc1Br Cc1ccc2c(c1)CCC2N(C)C(=O)Nc1ccc2c(c1)CCCS2(=O)=O Cc1ncc(NC(C23CC(NC(=O)C(C)O)(C2)C3)=O)c(C)n1 CCC(O)C(C)(C)C(=O)NCC(CC1CC1)C(=O)NC(c1ccncn1)C Cc1oc(C2CC2)nc1C(=O)NC1CCC(C)(CNC(=O)CCc2ccco2)C1 c1(C(=O)NC(C)C(=O)NCc2nc3sccn3c2C)cccc(C#CCO)c1 Cc1cccnc1C(=O)NCCCC(C)NC(=O)CNC(=O)CC1CCCC1 Cc1cccc2nc(N3CC=CC(NC(c4cc[nH]c5nccc4-5)=O)C3)oc12 N1(C(c2c(C)nc(C)[nH]2)=O)CCCC2(CCCN2C(=O)C(C)n2cccn2)C1 CC(C)C(C)(CNC(=O)CO)NC(C1CC1c1cnn(C)c1)=O C1(NC(c2n(CCC)ccc2)=O)CC(C(=O)N(CC(C)C)CCO)C12CCC2 C1(n2cc(C(CC)N(C)C)nn2)CCCN(C(=O)CCCc2nc(C)cs2)CC1 c1(C(=O)NC2CC(OC)CN(C(C3(F)CCC3)=O)C2)cc2ncccc2[nH]1 C(c1cnccn1)=CC(=O)NC1CC(C(CN(CCCC(=O)NC)C)=O)C1 c1(C(=O)NC(C(CO)NC(C(N2CC(C)C2)C)=O)C)cnc2ccccc2n1 C1(N(C(c2c[nH]c(=NC)o2)=O)C)CCc2cc(Br)ccc2C1 c1(N(CCCS(N)(=O)=O)C)nc(=NCc2cc[nH]n2)[nH]c2ccccc12 c1(C(=O)NC2CC(C(C(=O)NC(c3ncc[nH]3)C)F)C2)ccc(C2CC2)cc1 c1(C(=O)NCC(C)N(C(C(CC)C)=O)C)cc(C)nc2c(C)c(C)nn12 C1(C(=O)NC(CC=C)CNC(=O)C=CSC)OCCOC12CCC2 c1(CCCCC)ccc(C(=O)N(CCNC(=O)CCC2CC2)CCOCCO)o1 C12(NC(c3c(C)ncnc3C)=O)CCCC1CN(C(=O)CC1CCSCC1)C2 N1(C(c2cccc(NC(=O)NCCN3CCCCC3)c2)=O)CCc2ccc(F)cc21 N1(C(c2cc(CNC(CN3CC(C)(OC)C3)=O)no2)=O)CCCSCC1C C12(NC(c3cnc(C(C)C)[nH]3)=O)COC(CNC(=O)CN3CCCC3C)(C1)C2 C1(C(=O)NCC2CC(NC(C(N3CCCCC3)C)=O)C2)CCC2(CC2)C1 C12(NC(c3n(CC#N)ncc3)=O)CCN(C(=O)CCn3cncn3)CC1C2 c1(C(C(=O)NCC(CNC(C(CC)OC)=O)C)O)ccc(Br)cc1 S(=O)(=O)(c1ccc(C#N)c(N2CCOC(C)CC2)c1)N1CC(C#C)OCC1 CC1(CNC(c2c(Cl)nsc2Cl)=O)CCCN(C(c2cnn[nH]2)=O)C1 c1(NC(=O)NCC2CCCC2O)ccccc1-c1nc(C2CC2)no1 C=CC1(O)CCN(C(=O)C(C(C)O)NC(c2cncc(O)c2)=O)C1 c1(C(=O)NCC2CCC(NC(Cc3c(C)non3)=O)C2)cnc(N)c(Cl)c1 c1(C(=O)OC)nn(C)c(Cl)c1CN1CCC(C2CCCO2)C1 CC(C)CC(C(=O)N1CCCC(CO)CC1)ONC(=O)CCc1ccoc1 CC1(C)CCCC(C)(NC(=O)CCC2CCCN2C(=O)C=CCF)C1 C1(CC(=O)N(CC(C)OC)CC)CC2(C1)CN(C(C1C(=O)NN=C1C)=O)C2 C1(CNC(=O)CSCc2ccccn2)CCCC2(CN(C(C3CC3(Cl)Cl)=O)C2)O1 C1(NC(=O)CC)CN(C(=O)C(C)N(C)C)CC(C)(C)C1.N1(CCC)CCC(N)CC1 C1(CC(=O)NCCN(C(=O)COCCF)C(c2nccs2)C)C=CCCC1 c1(C(=O)NCCC2C(C)CN(C(C3CN(C(N)=O)C3)=O)C2)nn(C)cc1[N+](=O)[O-] Cc1ccccc1C=CC(N1CC=C(CNC(c2ncn(C)n2)=O)CC1)=O C1(NC(C(C)Cc2cnn(C)c2)=O)CC(F)CN(C(c2csc(C3CC3)n2)=O)C1 c1(C(N2CC(NC(CC(CC)O)=O)CC2(C)C)=O)nc2cc(F)ccc2s1 c1(C(=O)NC2CC3(CN(C(C4(C)CCCO4)=O)C3)C2)cc(O)c(F)cc1N c1(OC)ccc2ncccc2c1C(N1CCC(NC(c2cc(N)ccn2)=O)C1)=O c1(C(=O)OC)cncc(N2CCCC(NC(=O)NC3CC(C(N)=O)C3(C)C)C2)n1 C1(NC(C(F)OC)=O)CCN(CCNC(c2occc2-c2cnn(C)c2)=O)CC1 c12cccc(c1)CN2.Cn1cnc(CNC(c2cn(CCC3CC3)nn2)=O)n1 C1(C(=O)N(CC(F)(F)F)CCCOCC2CC2)CCOC2(CCOCC2)C1 N1(C(C2CC2F)=O)CC2(C1)CN(c1ccn3nccc3n1)CCO2 N1(CCC)CCCC1C(=O)N(CCC1(NC(C2C=CCC2)=O)CCC1)C(C)C N1(C(C2OCCC(C)C2)=O)CC(O)CCC1C(=O)NCCC1(C)CCCC1 N1(C(=O)NC2C(OC)CCC2)CCCC(Oc2ccc(F)cc2)C1 C(CCN=c1[nH]c(=NC2CC(NC(=O)NC3CC3)C2)[nH]c2c1CCC2)N(C)C C1(c2ccccc2)(NC(C=NOC)=O)CCN(C(=O)C(C2CCCOC2)OC)C1 N1(C(CCC#C)=O)CCC(C(=O)NC(C)CCC2CC2)CC1C CC1=C(C)CC(C(=O)NCC(C)(Cn2cccn2)NC(=O)CC(C)C(C)C)CC1 Cc1cc(CC(=O)NCC(F)CNC(=O)CCc2ncc[nH]2)n[nH]1 CC1(C(=O)NC2CCN(C(c3nnn4c3CSCC4)=O)C2)CC2(C1)CC(F)(F)C2 N1(C(CC2(C(=O)OCC)CC2)=O)CCC2CCN(C(=O)C=C(C)C3CC3)CC2C1 c1(C(N(C(CNC(=O)CC(O)C2CCCC2)C2CC2)C)=O)ccc(F)cc1 C(=O)(CCCC(=O)NCC(F)CNC(=O)CC1C(=O)N(C)N=C1C)NCC CCC(CC(F)(F)F)C(=O)N1CC(CNC(=O)CCCF)C2(CCC2)C1 C(=O)(C(=O)N=S(C)(C)=O)NC(C1CCCN1C(c1ccccc1C(F)F)=O)C N1(C(c2c(C(C)C)nco2)=O)CC2CC(NC(C3(CN(C)C)CC3)=O)C(C2)C1 c1(C(=O)NC(CNC(c2c(C)cn(-c3ccccc3)n2)=O)C)ccc(=O)n(C)c1 C1(CNC(CC=CC=C)=O)CN(C(=O)C=Cc2ccc(SC)s2)CC1(C)C C1(CC)(OC)CN(C(=O)C=CC(C)NC(C2(N(C)C)CC2)=O)C1 N1(C(CNC(CC)=O)=O)CC(NC(=O)C=Cc2cncnc2O)CC(C)C1 c1(C(N(CC=CC(=O)NCCC(CCC)C)C)=O)cccc(C)c1C#N N1(C(CN(C(C(C)C)=O)C)=O)CCC(C)(CCNC(C2CCN2S(C)(=O)=O)=O)C1 C(=O)(CCC(=O)c1ccccc1N)N(CC(C)CNC(=O)CNC(=O)C1CC1)C C=CCC(C)(C)CC(=O)N(C1CN(C(=O)CCCn2cncn2)CCC1O)C c1(OC)nc(N2CCC(c3cc(O)no3)CC2)cnc1Br Cc1cc(C(N2CCCC2C(C)NC(=O)COc2ccc(F)cc2)=O)cc(F)c1 Cc1cc(O)ccc1C(=O)N(C1CCN(C(=O)CC(C)(F)F)CC1)C c1(CC)cc(O)nc(-c2cccc(NC(c3cn(C(C)C)nn3)=O)c2)n1 N1(C(=O)NCc2coc(O)n2)CCCC(O)(C2CC2)C1 CC1(C)CCC(C(=O)NC(Cc2cnc[nH]2)C(=O)NC2CNC(=O)C2(C)C)CC1 C1(NC(C(C(=O)OC)OC)=O)CC(C(N2CC(O)CC(O)C2)=O)C12CCC2 N1(C(C(C)=CC)=O)CCC(C)(C(C)(C)NC(=O)CCC=Cc2ccccc2)CC1 Cc1ccc(C(c2nnnn2C2(C)CC2)NCc2ccccc2C)cc1 N#CC1CCCCC1NC(C1CCC(CNC(C2CCOC2)=O)C1)=O C1(CNC(c2cccc(OC(F)F)c2)=O)CN(C(=O)CSc2nncs2)C2CC12 CC1COc2ccc(C(N3CCC(NC(C4CN(C)C4)=O)C3C3CC3)=O)cc21 c1(CC(=O)OC)cccc(N(C)C(C2C3CCC2(c2cccs2)C3)=O)c1 C(=O)(C(C)C(O)C(C)CC)N1CC(C(C)(C)O)(CNC(CC(C=C)(C)C)=O)C1 N1(C(c2nc(C(C)C)oc2)=O)CC(C)C(N=c2ccc(C#N)c[nH]2)C1 C1(NC(C(C)=C2CC2)=O)CCC2(CC1)CN(C(=O)C(F)CC(C)(C)C)C2 c1(C(N2CCC3CN(C(C(C)SCCCC)=O)CC32)=O)cc2nc[nH]c2cc1N CC1CC(C(=O)NC2CN(C(c3cc(C4CCC4)on3)=O)C2)CC(C)O1 c1(C(=O)NCC(C)CNC(C2CCCC2F)=O)cc(Cl)c(Br)cc1F N1(C(=O)CCC2CCC2)CC2CC(NC(=O)C(c3ccc(F)cc3)(F)F)CC1C2 n1(CCN(C(=O)CCNS(C)(=O)=O)CC)cc(CC2(O)CCSC2)nn1 C12(NC(C=CC(=O)N(C)C)=O)COCCC1CN(CC1(N3CCCCC3)CC1)C2 c1(OCC=C)ccccc1C(=O)NCC1CCCC(NC(c2coc(O)n2)=O)C1 C1(NC(c2c(C)n(C(C)C)cc2)=O)C2CC1N(C(=O)C(c1ccccc1)F)C2C C(=O)(CCS(N)(=O)=O)N(C1CCN(c2nnn(C)n2)C1)CCC C1(C(C)C(=O)NC2(c3nn[nH]n3)CC2)CCN(C(=O)C(=O)C2CCCC2)C1 C(=O)(C(C)(C)C(=O)N1CC2C(CN(C)C(c3cnccc3Cl)=O)C2C1)NC C12(NC(c3ccnc(C)c3C)=O)CCOCC1CN(C(=O)Cc1cnn(C)c1)C2 C1(C(=O)NC2CCC(CNC(CNC(C)=O)=O)C2)CCc2nn[nH]c2C1 N1(C(C(=O)NCC)=O)CCC(n2cc(CNC(=O)C(C)OCC(C)C)nn2)CC1 C12(C(=O)NC3CCCC(NC(CCCC=C)=O)C3)C3C4C1C1C2C3C41C c1(C(=O)NCC2(O)CN(C)C2)cccc(CNC(=O)Cn2cccn2)n1 c1(C(N2CCN(C(C(C)O)=O)C(CC(F)F)C2)=O)cc2c(F)cc(F)cc2[nH]1 N1(C(C2CN(NC(C(=O)C(C(C)NC(=O)C3CC3)=O)(C)C)C2)=O)CC2CCC1C2 C1(F)(C(N2CC(CC(C#C)C)C2)=O)CCCN(C(C2CCC(=C)CC2)=O)C1 C(CS(=O)(=O)c1cnn(C)c1)NC(=NCCCC)NCC(CO)C1CCOC1 C(Cc1ccccc1)(CCNC(C1CC(N(C)C)C1)=O)NC(COCC(=C)C)=O C1(C(N(CCC(=O)OC)C)=O)CC12CCN(C(C1(O)CCSC1)=O)C2 N1(C(C(N2CCC(CC#N)C(F)(F)CC2)=O)=O)CCCC2(CC=CCC2)C1 N1(CCNC(=O)C(N)C2COC2)CCN(CCN2CCCC2)CC1 c1(C(N(C2CCN(C(CCN(CCCCC)C)=O)C2)CC)=O)ccc(O)c(N)n1 CC1CC(C)N(C(c2cn(C)c(O)n2)=O)CCN1C(=O)CCSCc1ccncc1 C1(NC(c2n(C(C)C)ccc2)=O)CN(C(=O)CCC(C)(C)C)CCC1(C)C C(CC(C(C)C)NC(c1nocc1C(C)C)=O)NC(C=C(C)C1CC1)=O C(=O)(C1=C(C)CCC1)NC1(C(N(CC)CC2CCC2)=O)CCCC1C c1(C(N(CCOCCC(=O)N(c2cccc(O)c2)CC)C)=O)ncc(F)cc1C C1(NC(Cc2cn(CC)nn2)=O)CCN(C(C2(C)CCN(C)C2)=O)C(C)(C)C1 n1(C(C)C)nnnc1C(CCc1ccsc1)NCc1ccc(-c2ccccc2)s1 C(=O)(C1c2c[nH]nc2CCC1C)NCCOCCCNC(c1cc(C)[nH]c1C)=O C1(CF)CCN(c2cc(N3CCC(C4CCCCO4)CC3)ncn2)CC1 N1(C(c2ccn(CC)c2C)=O)CCCC2(C1)CN(C(C1CC1C)=O)CCO2 O(N1CCC(NC(=O)CCCC(C)NC(C2CCC(C)(O)CC2)=O)CC1)CC c1(N2CCC(C(C)(C)C)(CNC(Cn3c(=N)scc3)=O)C2)ccc([N+](=O)[O-])cc1 CC1C(=O)CCC(C(=O)NCCCc2ccc(-c3nn[nH]n3)cc2)C1(C)C C1(C(=O)NCC(N(C(=O)CC2CCCC(=O)N2)C)C2CC2)CC(=O)CC12CCC2 c1(C(=O)NCCC(=O)NCC(O)CNC(C2CC23CC3)=O)cn2ccccc2n1 c1(C2CCCN(C(c3ccc(-c4ccncc4)cc3)=O)C2)cccc2cc[nH]c12 c1(C(N2CC(C(=O)NC3(C#C)CCOC3)C(OC)C2)=O)cccc(C#N)c1C C(=O)(C1=CCOCC1)N1CC(CO)C1.C(C1C(=O)N1)C(C)=O.C(C)(C)(C)OC(C)=O C1(N(C(C2N(C)C(=O)NC2)=O)C)CN(C(C2CC(Cl)(Cl)C2)=O)CC12CC2 N1(C(c2c(SC)c(F)ccc2)=O)CCCCC1C1CCCN1c1ncccn1 c1(C(N(C)C)=O)cn(CC(=O)NC2CCC(NC(c3cnnn3C)=O)C2)nn1 C1(CCC)CN(C(c2cnn(C)c2SC)=O)CCN1C(c1cc(C)c[nH]1)=O N#CC1(C(=O)NCC2(F)CC(NC(=O)Cn3cnccc3=O)C2)CC=CC1 Cc1cccc([N+](=O)[O-])c1NCCCNC(=O)Cn1cc(C2CC2)nn1 c1(CN(C(C(C2CCCC2)NC(C(SC)SC)=O)=O)C)cccc(O)n1 N1(C(CN(C(CCNC(=O)OC)=O)CCO)=O)CC(O)CC(O)C1 C(C)(CC(=O)NCCOCCC(=O)N(C(C)C)Cc1cn(C)cn1)SC C(C(CNC(=O)CC1CCCCCC1)C(F)(F)F)NC(C(C1CC1)SC)=O S(=O)(=O)(c1cc(F)ccc1F)NC1C(C(=O)NCc2cscn2)C1 C(=O)(C1=CSCCO1)N(CC(C)NC(=O)CN1CCCC(N(C)C)C1)C c1(CC(=O)NCC(C)(C)NC(=O)C(c2ccccc2)NC(N)=O)cncc(F)c1 C(=O)(C1CC(=O)Nc2ccccc21)NCC1C(OC)CCC1 CC1C(NC(c2cnns2)=O)CCN1C(=O)CCC1CC1(Cl)Cl C(=O)(C1=NOC2COCC12)NC1C(C(N(C2CCCC(C)C2C)C)=O)CCC1 N1(C(CNC(=O)OCC=C)=O)CCCN(C(=O)Cc2cc(C)ccc2C)CCC1 C1(NC(c2n(C)nc(C(F)F)c2)=O)COC2(C1)CN(C(c1csc(S)n1)=O)C2 C1(N(C(Cn2c(N)ccn2)=O)CC2CCOCC2)CCN(c2cccnn2)CC1 C(=O)(C#CC1(C)CCCO1)NC(CNC(C=C(CCC)C)=O)C(C)C c1(C(=O)NCC(C)N(C(c2cc(Br)n(C)n2)=O)CC)cccc2c1OCC2 C(=O)(CC(C(C)CC)NC(=O)C(CCC)NC(C)=O)NCC(CC#C)(C)CO CCC(CC)(CC)S(=O)(=O)CCOc1ccc(F)cc1Cl CON=CC(=O)NCCC(C)N(C)C(c1cnc(C(C)(C)OC)s1)=O N1(C(C2(CCC=C)CCCC2)=O)CCC(C(F)F)(CNC(=O)CSC2CC2)C1 CC1(C)CN(C(=O)CS(=O)(=O)NC2CC2)CCC1NC(=O)CCC(N)=O CC(O)C(O)CNC(=O)C(C1(O)CCC1)NC(=O)CC1(O)CCOC1 C1(CNC(=O)NCCc2nc(CC)on2)(OC)CCOC1(C)C C(CO)(C(F)(F)F)NC(CC1CCN(C(C2C(=C)C2)=O)C1)=O C12(NC(C(C)c3ccco3)=O)CC(CNC(=O)Cn3cccn3)(C1)OC2(C)C C1(CNC(c2c(CC)n(C)nn2)=O)C(O)C(O)CN1C(=O)CC1CCCC1OC C1(NC(c2[nH]cc(CC)c2)=O)C2CCN(C(c3c[nH]c(=N)nc3CC)=O)CCC12 c1(C(=O)NC2C(CNC(C(C3CCC(=O)N3)C)=O)C2)ccc(NCCO)cc1 c1(C(=O)NCC2CCCN2C(=O)C(F)=CCCF)ccc(F)c2cccnc12 c1(C(N2CCC(NC(C3(C#N)C(C)(C)C3)=O)C(O)C2)=O)ccc(F)cc1C#N N1(C(C2N(C(c3ccc(C(C)=O)o3)=O)CCSC2)=O)CCC2(C1)CC2(F)F C1(NC(Cc2nc(C)sc2)=O)CCOC(C(=O)NCCCc2ccco2)C1 CN=c1[nH]cc(C(=O)NC2CN(C(c3cnsn3)=O)CC2c2cccc(F)c2)s1 CC(CNC(C12CCCC1C2)=O)C(=O)NC(C)C(=O)NO C12(CN(C(c3c(C(N4CC(C)C4)=O)cccc3)=O)C)C3C(=O)C4C5CC(C14)C2C35 O=C1CCC(C(=O)OCC(C2CC2[N+](=O)[O-])=O)=NN1 C(C)(CNC(=O)CN1CCCC1)(CNC(=O)CC1(n2ccnc2)CC1)OC c1(C(=O)NC(C2CCCCC2)C(C)NC(CC)=O)cc(C)cc(OC)c1C N1(C(c2cc(Cl)cnc2O)=O)CC2CCC(C1CO)N2C(=O)C(O)CC1CC1 c1(C(C(=O)NCC(c2nncn2C)C)(C)C)c[nH]c2cc(F)ccc12 CCC(C)CCCC(=O)NC1CCCCC1NC(=O)CCn1nc(C)cc1C C(CC)(C(=O)N(CC(=O)NCCCOCCCC)C1CC1)=CC N1(CCOC)CCCC(NC(=O)COc2ccc(OC(F)(F)F)cc2)C1C C1(CCNC(CC)=O)COCCN1C(c1ccc(OCF)cc1)=O.C1C(=O)O1 c1(CC)nc(C)ccc1CNC(NCC1=C(C)OCCS1)=NCCc1ccsc1 N1(C(Cc2ccc(C)s2)=O)CCN(C)C(CNC(=O)Cc2cnco2)C1 N1(C(C(C(=C)C)(C)C)=O)CCC2(CCC2CNC(=O)Cc2cc(C)cs2)CC1 c1(C(N2CC(CNC(=O)C(=O)NC3CC3)C3C2C3)=O)cccc2c1OCCN2 c1(CC(=O)NC2(C)CC(NC(c3c[nH]c(C(N)=O)c3)=O)C2)cnc2n1CCOC2 Cc1ccc2c(c1)C(Nc1nccc3occc13)C(C)C2 c1(C(N2CCCCC2CC(F)(F)F)C(=O)NC(CC)C)ccnc(OC)c1F N1(c2nccc(CC(=O)OC)n2)CC2CC(NC(=O)C(C)SC)C2C1 c1(CC)ccc(NC(C2CSCN2C(=O)CNC(=O)C(C)(C)C)=O)cc1C N1(C(c2c(C(C)C)c[nH]c2)=O)CC(NC(=O)CCc2nc(=N)[nH][nH]2)CC(O)C1 C12(NC(C(CC=CC)NC(C3CCOC(C)(C)C3)=O)=O)CCC(O)(CC1)CC2 CCCCC(=O)NCCN(C1CCCC1)C(=O)CNC(=O)Cc1nncn1CC n1(CC)cc(CCC(=O)N(C2CN(C(C3C=C(C)CS3)=O)C2)C)cn1 C=CCC(C)N=c1[nH]c(=NC(COC)CCO)[nH]c2cccnc12 C#CC1CN(C(=O)C(C)n2cccc2)CCN1C(=O)CC(C)n1cccc1 C1(C(=O)NCc2ncc(C(=O)NC(C3(OC)CCC3)C)cn2)CCOC(=O)CC1 CC12CC3CC(C(=O)NC4CC(NC(=O)CCc5ccsc5)C4)(C1)CC(C)(C3)C2 c1(OC)c(CC(=O)NCC2CCCCN2C(=O)C=CCO)cccc1F N1(C(CCN(CC)CC)=O)CCN(C(=O)C=C(C)C(C)C)CC(C)(F)C1 C1(CNC(CC(CCC)C)=O)CCC2(CN(C(=O)CCC3CC3)C2)O1 C(=O)(CC1CCc2ccccc21)NC1CC(CNC(CCS(=O)(=O)N(C)C)=O)C1 C1(C)(CC)CCCC(NC(=O)CCn2cc(-c3cc(C)cnc3F)nn2)C1 N1(C(C(C)SC)=O)CCN(C(c2ccc(CC3CCC3)cc2)=O)C(CF)C1 N1(C(c2c(CCC)snn2)=O)CC2(CC(n3cc(C(=O)OCC)nn3)C2)C1 C12(C(=O)NC3CN(C)C3)CC(n3cc(C(C)(C)NC(C)(C)C)nn3)C1C2 c1(C(=O)NCC(C)N(C)C(C23CCCC(CO2)C3)=O)ccc2c(n1)NCCO2 C1(NC(c2cncc(N(C)C)c2)=O)CCN(C(c2ccc(CO)s2)=O)CC1F C1(CNC(C2C(Cl)(C(=O)OCC)C2)=O)(NC(=O)Cc2ccccn2)CCCCC1 N1(CC(=O)NC2(c3ccc(Br)cc3)CC2)CCS(=O)(=O)CC1.c12cn(nn1)C2 CC1CCc2[nH]c(C(=O)NCCC(C)(C)S(C)(=O)=O)cc2C1 c1(C(N2CCN(C(C3CCOC3)=O)CC2)C(=O)NC)cc(Br)c(C)nc1OC C1(C(N(C(CC)CC)CC)=O)C2CN(C(C)Cn3cc(C)cn3)CC12 C1(c2ccccc2)(NC(c2csnn2)=O)CCN(C(=O)CC2CCCO2)CC1 C1(NC(CC2CC(=C)C2)=O)CC(C)N(C(c2ccc(CCCC)cc2)=O)C1 Cc1cc(C(=O)NCC2CN(C(=O)C3=CCCC3C)CCO2)cn(C)c1=O C(C(=O)N(CC(=O)NC(COC)CO)CC)(C1CC1)OCC N1(C(c2n(C)[nH]c(=N)c2)=O)CC(F)(F)CC1CNC(c1c[nH]nc1[N+](=O)[O-])=O C(CC(C)C)(C(=O)NCCc1cnco1)NC(C(C1CCC1)OCC)=O C1(NC(c2ccc(C(C)(C)C)[nH]2)=O)CN(Cc2ccc(CBr)cc2)CC1F C1(N(C(=O)C(C)CNC(C2CC2CCC)=O)CC#C)CCN(C(C)=O)CC1 C(=O)(C1=CC(C)(C)C1)N(C(C)C(=O)N(CCCC(C)(F)F)C)C N1(C(C2(COC)CC2)=O)CC2CCC1C2NC(=O)CCC(C)SC c1(C(=O)NC2CC(F)(CNC(C(C)NC(C)=O)=O)C2)ccc2nn[nH]c2c1 CCCCC(CC)CC(=O)NCC(C(=O)NC1CC(N(C)C)C1)N(C)C c1(C(N(C(CNC(C2CCCC3(CC3)C2)=O)C2CC2)C)=O)cc2ncccc2o1 c1(C(=O)NC(CNC(C(C)NC(CC)=O)=O)CC)ccc(C#N)nc1C Cc1nc(C(=O)NC2CCC2NC(C2CC(=O)N(C(C)C)C2)=O)ccc1Br C(C(=O)N=c1cc(C2CCOCC2)[nH][nH]1)c1cccc(C(=O)O)c1F Cc1cc(C(=O)N(C(C)C(=O)Nc2ccc(Cl)nc2)C2CC2)ncn1 C1(C2CCN(C(c3cscc3Cl)=O)CC2)(NC(C2CCC2(F)F)=O)CC1 Cc1oc(Br)cc1C(N1CCCC(C(C)NC(C2(N=[N+]=[N-])CC2)=O)C1)=O C1(C(=O)NC2CC(C)(NC(=O)CSC3CC3)C2)CCc2ccnn2C1 N1(C(c2ncn(CC)c2)=O)CC(C)CCC1CNC(C1(C(F)F)CCC1)=O c1(C(=O)NCC2C(NC(c3c(CC)noc3)=O)CCC2)cc(OC)cc(CC)c1 CC1(C)C2CCC(C(=O)NCC3CCN3C(=O)C(C3CCOCC3)F)C1C2 N1(C(C2C(CC)C2)=O)CCN(C)C(CNC(=O)COC(F)(F)F)C1 c1(C(N2CC(CNC(c3cc(CCC)[nH]n3)=O)C2)=O)ccc(OCC)c(Cl)c1 CC1(C2CCN(C(C3CCN3C(C3C4CCC(F)C34)=O)=O)C2)CC1 c1(C(N2CC3C(CC(N4CC(CC)N(C)CC4)=O)(CC3)C2)=O)ncc(C#N)cc1C c1(CC)cccc(C(=O)NC(C)(CNC(C2CC(C(C)C)=NO2)=O)CO)c1N c1(OC)ccc(C(C)C(=O)NCC2CCN(C(=O)C3=C(Cl)CC3)C(C)C2)c(C)c1 N1(c2nccc(=NCc3ccc(CC)s3)[nH]2)CCc2c(F)cccc2C1 C12(NC(C(C)C3CCOC3)=O)CC(C(=O)NCC3CCC(O)C3)(C1)C2 c1(C(=O)NCCN(C(=O)Cc2ccsc2)CCC)ccc(CNC(C)=O)s1 C1(NC(CN(CC)CC)=O)(CO)CN(C(=O)CC(C)C2CCCO2)C1 Cc1cccc(C2CCCN2Cc2cn(CCO)nc2-c2ccccc2)n1 C(C(CC(C)C)C(=O)N1Cc2cncnc2C1)NC(c1nccc(CC)c1)=O c1(C(N2CCCC2C2CC2(F)F)C(=O)NC(C(=O)OC)C)cc(C)cs1 N1(C(C2(OC)CCOC2)=O)CC2(CC(NC(=O)CCCF)c3nccn32)C1 C1(C(=O)NC2CC(CNC(c3onc(CC)c3C)=O)C2(C)C)CN2CCN1CC2 CC1CC(NC(c2ccc(CO)c(F)c2)=O)CN(C(c2cc(F)ccc2Cl)=O)C1 C1(NC(=O)CCCCCF)CC1C1CCN(C(=O)CC2CCCS(=O)(=O)C2)CC1 N1(C(c2c(CC)c[nH]c2)=O)CCN(C(C2CSCN2C(C)=O)=O)C(CO)C1 C1(CNC(C(CC)C)=O)CN(C(C2(c3cccc(Cl)c3)CC2)=O)CC1C C1(NC(c2nc(CCC)sc2)=O)CN(C(=O)C(C)=C(C)CC)C2(CCC2)C1 CCC(C(=O)NCCN(C)C(C1(Br)CC1(C)C)=O)c1ccccc1 C1(NC(C2(C(=O)NC)CC2)=O)CCCN(C(=O)C(C)OCC(C)C)CC1 Cc1cc(C(=O)NC2CCN(C(C)C(=O)NCc3cccs3)C2)c(C)[nH]1 C1(NC(C23N(C(C(O)NC(=O)OC)=O)CC(C2)C3)=O)CC2(CCCCCC2)C1 C1(CNC(c2c(C)cn(C)n2)=O)CC(NC(=O)Cc2cncs2)C12CCC2 CC#CCC(C(=O)NC(CO)C1(O)CC1)NC(c1cc(C(C)=O)c[nH]1)=O N1(C(CNS(NC)(=O)=O)=O)CCC2(CC2NC(=O)CC2CCC(C)(C)C2)C1 c1(C(N2CC3C(CNC(c4cc(Cl)cs4)=O)C3C2)=O)ccc2nnc(S)n2c1 c1(C(N(C)CC2(O)CN(C(C(F)=C(C)C)=O)C2)=O)cncc(F)c1C c1(CC)nc(-c2nc[nH]n2)sc1C(=O)NCC1CC1NC(c1oncc1C)=O C12(CNC(C(CC3CC3)OC)=O)CC1CN(C(=O)CN1CCC(N(C)C)CC1)C2 C1(OC)(OC)CC(C)(C(N2CC(CCCCNC(C34CC(C)C3C4)=O)C2)=O)C1 C1(COC)CC(CNC(C2CC(C)(C)CO2)=O)N(C(c2occc2C2CC2)=O)C1 C1(CNC(CNC(CCC)=O)=O)CC2CCC1N2C(=O)CCc1cnn(C)c1C N1(C(c2ccc(C#N)[nH]2)=O)CC2CCN(C(c3n[nH]c4c3CSCC4)=O)CC12 N1(C(C(CC)=CCCC)=O)CCC(NC(c2cccc(C3CC3)n2)=O)C12CC2 N1(C(=O)Nc2cnc(C(F)F)nc2)CC(n2cccn2)Cc2ccccc21 C1(C(=O)NCC(CNC(c2ccc3ncnn3n2)=O)O)CCCC12CCOCC2 C(CCCCC(=O)N1CCCC1c1cccc(C)n1)NC(c1c(CC)non1)=O CC(C)(CCC(=O)NC1CC(OCC(=O)NCC2CNC(=O)CO2)C1)[N+](=O)[O-] Cn1nc(C(=O)NCC2CCN(C(=O)C=CC(=O)NC3CC3)CC2)c(Br)n1 c1(CCC(=O)N(C)CC2(NC(C3CC3Cl)=O)CC2)cccc(Br)c1Cl C(CC(F)F)(C(=O)N1CC(C)C1(C)C)N(C(=O)CC12CCC(CC1)C2)C c1(C(N2C(C)CCC(CNC(=O)C3=CCCC3)C2)=O)cccc2c1CCC(=O)N2 c1(OC)nn(C)nc1COC(c1nnn(Cc2cc(C)on2)c1C)=O C(=O)(C(C)CC(C)(F)F)NCC(CC)(CC)NC(c1cccc(S(C)=O)c1)=O C12(C(=O)NCC3C(CNC(c4cn(CCO)nn4)=O)C3)CCC(=O)N1CCS2 c1(NC(C(C)C2CCCO2)=O)cccc2c1NC(=O)CC2 c1(C(N2C(C(=O)NCCN(C3CCCC3)C)CCC2C)=O)cc(C)cc(O)c1 N1(C(c2cc(CCC)on2)=O)CCC2CC12C(=O)NCc1cc(C(N)=O)co1 C1(C(=O)NCC(CC)NC(c2[nH]nnc2C2CC2)=O)CC(C)(C)C1C(F)(F)F N1(C(C(C)OCc2cccc(C)c2)=O)CC2(C1)CN(C(=O)C=CC(=O)N(C)C)C2 CCC(CCC(=O)NCC(C1CCC1)NC(c1csnc1OC)=O)OC c1(NC(C(CC2CCCC2)NC(COCCC#C)=O)=O)cncc(C2CC2)c1 C1(C(=O)NCC(n2cncn2)C)CCN(C(c2ncccn2)=O)CC1 N1(C(c2ccc(C)s2)=O)CCC(O)(C(C)NC(=O)CCc2nnc(C3CC3)o2)C1 c1(OC)cnc(CNC(=O)C(C2(C)CC2)NC(C2CCC(=O)C2)=O)cn1 Cc1noc(C)c1C(C)(C)C(=O)N1CCC(N(C)C(C2CCCC(F)C2)=O)C1 C(=O)(C1=CCCCCC1)N1C(C)CN(C(=O)CCOc2ccc(Br)cc2)CC1 c1(CN2C(C(=O)NCc3ccc(C(F)F)nc3)COCC2)cc(Cl)c(Cl)cc1Cl c1(OC)cccc2c1CN(C(C1CC1c1cccc(-c3ccoc3)c1)=O)C2 CCCC(C)CC(=O)N1CCOC(CN(C)C(c2cc(CC)n(C)n2)=O)C1 C1(NC(c2n(C)ccc2)=O)CC(O)CN(C(=O)CCCc2ccc(Cl)cc2)C1 N1(C(COCC)=O)CCCC(O)(CNC(C2(C)COC(=O)C2)=O)C1 c1(CC(=O)NCCCC(C)O)ccc(-c2ccncc2F)c(F)c1 N1(C(C(C)Oc2ccccc2)=O)CC2CCC1C2NC(=O)CC(C)C(F)F c1(C(=O)NC2C(OC)CN(C(c3cnn(C)c3F)=O)C2)ncc(N)cc1Cl c1(OC)cc(Br)ccc1CN1CCC(C)(C(=O)N(CC(F)(F)F)C)CC1 c1(OC)ccc(C)cc1C(N1CC(O)CC1C)C(=O)NCCC1CC1 c1ccc2c(c1)CCSC2Cc1nc(-c2cnc3c(c2)OCO3)no1 c1(CC(N2C(C(C)NC(C3SCCS3)=O)CCC2)=O)ccc(F)cc1F Cc1cc(C(=O)NC(C)C(CO)NC(=O)C=CC2CCOCC2)nnc1O c1(CN=c2sc3c([nH]2)C(=O)CCC3)nc(O)c2ccc(C(F)(F)F)cc2n1 N1(C(COCCOCC)=O)CCC(F)(C(N2CC(OC(C)=O)C2)=O)CC1 c1(C(=O)NC2CN(C(c3cnn(CCC)c3C)=O)CC2C)n[nH]c2c1CC1CC21 C1(CNC(C(CC=C)NC(C)=O)=O)CN(C(=O)CCCOCC)CC1(C)C C1(CCNC(C2ON=C(C)C2C)=O)CCN(C(c2ccc(SC)o2)=O)CC1(F)F C(CCC(C)(C)C(=O)NC1CCCCC1CNC(=O)C(C)=CC(C)(C)C)OC CC(C)(C)CC(O)C(=O)NCC1(O)CCCN(C(=O)CCc2ccccn2)CC1 N1(C(CCCCC)=O)CCC(C2CCCN(C(=O)C(C)(C)C(C)(F)F)C2)C1 C1(CC)CN(C(=O)OC(C)(C)C)CCC1NC(c1c(C)nnn1C(=O)O)=O c1(CNC(C(C2CC2)OC)=O)ncoc1CCNC(C1CC(C(F)(F)F)C1)=O C1(=CCNC(=O)C(CO)c2ccccc2)CCN(C(=O)C(F)(F)CO)CC1 c1(CC(N2CCCC(CCNC(=O)C=CCBr)C2)=O)cc(Cl)ccc1Cl C1(NC(CCOC)=O)CCC2(CCCN(C(C3SCC=C3C)=O)C2)C1 c1(C(N2C(CNC(C3CCCSC3)=O)CCC2)=O)ccc(N2CCC2)nc1 N(C1CCCc2c(Br)cccc21)CC1(C)NC(=O)NC1=O N1(C(CC(CC)C2CC2)=O)CC(NC(=O)C(c2ccc(C)cc2)F)CC1(C)C CCCCCCCCC(=O)NC1CC(C(=O)NC(c2ncn(C)n2)C)C1 Cc1ccsc1C1(C(=O)NC2(C)CC(C)C2)C(NC(=O)C2CC2)C1.C(C)C CCCC(CNC(=O)CCCc1ccccc1)NC(=O)Cc1ncc(C)s1 c1(C(=O)NCC2N(C(CS(CC)=O)=O)CCCC2)ccc2c(n1)CCCN2 C(=O)(C(F)CC(C)(C)NC(=O)C(O)CCC(C)C)NCc1nnc(C)s1 N1(C(C=CC(=O)NCC)=O)CCC(NC(=O)COCCCF)CC1 c1(C(N2C(CNC(CC)=O)CC(O)C2)=O)cc(OC(F)(F)F)ccc1Br c1(C(N2CCN(C(=O)CCCn3cccn3)C(C3CC3)C2)=O)ncc(F)cc1F n1(CCOCCCOCCCO)cc(NC(C2(CCSC)CCC2)=O)nn1 c1(C(C(=O)NC2CC2)N(c2ccc(C)cc2)CCCC)nn(C)c(C)c1Cl c1(OC)ccc(CC(N2CCC(CN(C(=O)C=C(C)C(C)C)C)C2)=O)c(C)c1 N1(C(c2ccc(COC(C)C)nc2)=O)CCCN(C(=O)C(C)(C)C2CC2)CC1 C1(COC)(CNC(C2(C)CC2(C)C)=O)CCN(C(C2CCN(C)CC2)=O)C1 C1(CCNC(C2COC(=O)O2)=O)CCCN(C(=O)Cc2cc[nH]c2)C1 c1(C(=O)NC(CC=C)CNC(=O)CN2CCC(CC3CC3)CC2)ccc(Cl)cc1 Cc1ncccc1NC(C1CC2CC2N1C(=O)CC1CCCN(C)C1)=O c1(CCCNC(C2(NC(c3ccccc3F)=O)CC2)=O)c(F)cccc1Cl c1(N2CCC(C(=O)OC)C(OCC)C2)nc2c(cc1C#N)C=CC1(CCCCC1)O2 C1(CNC(=O)CNC(c2ccc(F)cc2)=O)CN2CCCCC2CO1 N1(CC)CC(CNC(=O)C(=O)NC(c2c(C)noc2C)C)CC1=O N1(C(CC2C(CNC(C=CC(C)C)=O)C2)=O)CCCC1(C)C CC(C)C1C(=O)O1.c1(C2CC(C(=O)Nc3ccccc3)C2)ccccc1Cl c1(CNc2c(C(=O)NCC3CN(C)C(=O)C3)n[nH]c2)c(F)ccc2occc12 Cc1ncc2n1CCC(C(=O)OCc1ccc(CC#N)cc1)C2 C12(NC(C3CCCCN3C(c3cncc(CO)c3)=O)=O)CCN(CC1)C2 c1(C(=O)NC2CN(C(C3(CC)CCCC3)=O)CC2C)cc(Cl)ccc1OC(F)F N1(C(=O)Cc2ncc(Cl)s2)CC2(CCN(C(=O)CC3CC4CC4C3)C2)C1 C1(C(N(CC(N2CCCC2)C)C)=O)CC=CCC1NC(=O)COCCCN=[N+]=[N-] c1(C(=O)OCc2c[nH]cc2C(F)(F)F)ccc(I)c(OC(F)(F)F)c1 c1(CCC(=O)NCC(n2cc(C(C)(C)CO)nn2)C)ccc(C(=O)N(C)C)cc1 c1(CN2CCC(F)(C(=O)Nc3ccc(OC)c(I)c3)C2)c[nH]c2ncc(Br)cc12 N1(C(C(c2ccc(Cl)cc2)C)=O)CCN(C(c2cc(C#N)on2)=O)CC(O)C1 C(=O)(CC(C(F)(F)F)N1CCOCC1)NC1C2C(C)N(C(=O)C=C3CCC3)C1C2 C=CC1CN(C(=O)C(Cc2ccco2)NC(C2CC2C(C)(C)C)=O)CCO1 C(=O)(C(C)(C)CCOC)N1CCCC(CCCCNC(COCC(=O)OC)=O)C1 c1(C(=O)NCC(C)N(C(Cc2ncc(C)o2)=O)C)ccc(Cl)c(Cl)c1 N1(C(c2c(CC)n(C)cc2)=O)CCC2(CC1)CCN(C(C1CC=CCC1)=O)C2 c1(C(N(C)CC2N(C(C=CCC)=O)CCC2)=O)ccc(N)c(-c2nccs2)c1 C1(C(=O)NCC23CC(NC(c4c(C)cncc4)=O)(C2)C3)CCOCC12CCCC2 c1(OC)ccc(C(N2CCC(N(C(C3CC4(CCC4)CO3)=O)CC)C2)=O)c(C)c1 c1(CC(N2C(C(C)NC(=O)Cc3cnsc3)CCC2)=O)ccc2nonc2c1 C1(NC(C2N(C)CCCC2)=O)CC2CC(NC(c3ccnn3C3CC3)=O)C2C1 C=CC1(C(=O)Nc2cncc(F)c2)CCN(C(C2CCOC2)=O)CC1 N1(C(c2cc(C(C)C)no2)=O)CCC(CF)(NC(=O)C(C)Oc2ccccc2)C1 CCS(=O)(=O)c1cccnc1C(N1CC(NC(c2cnc(Cl)s2)=O)C(O)C1)=O C(=O)(C1=CC2(CN(C(=O)CSC(F)(F)F)C2)OC1)NC1C2CC(=O)OC2C1 CCC(C)(C(=O)NCC1(NC(=O)CCc2cnc(C)s2)CCC1)C(F)F C=CC(C)(C)C(=O)N(CC(CO)(CO)NC(=O)Cc1ncc(C)s1)C CC1CCN(C(c2cnn(CC(F)(F)F)c2)=O)CC1CNc1ccc(C#N)nc1 n1(CC(=O)NC2(CCC(=O)OCC)CCC2)ncc(C#N)c1N C1(C(=O)NCc2nc(CNC(c3ncc(N)nc3)=O)sc2)CCN2CCCC2C1 C(=O)(C1=CCN(C(c2nccs2)=O)CC1)NC1C(C)(C)CC1 Cc1cc(O)ncc1NC(C12CC1CN(C(=O)CCN1CCCC1)C2)=O N1(C(c2c(C)nn(C)c2)=O)CCCC(C)C1CNC(=O)C(C)NC=O N1(C(C=CC=CC)=O)CCC2CCCN(C(=O)CCn3ccnn3)C2C1 C12CCCN(C1)CC(=O)N1CC(C(O)C1)CNC(=O)C=CC2.C1(N)CCCCC1.CC N1(C(Cc2cc(C)on2)=O)CCC(CNC(=O)COC2(C)CCC2)(OC)C1 c1(CC)ccccc1OCCC(N1CCCC1CCNC(=O)CC1CCCO1)=O c1(C(=O)OCC)ccc2nc(CCNC(=O)C=Cc3ncco3)[nH]c2c1 C1(CNC(Cc2cc(C)nn2C)=O)C(C2CC2)CCN1C(=O)CCC1CCCC1 C1(C)(CC=C)CN(C(=O)C(C2CCN(C(=O)CN3CCCC3)C2)F)C1 N1(C(C2(C#N)CCC2)=O)CCC2(CCC2NC(c2snc(Cl)c2Cl)=O)CC1 c1(C(N2C(CCC(=O)OC(C(=O)NC)C)CCC2)=O)ccc(C2CC2)c(C)c1 C1(NC(c2ccc(C)cn2)=O)CCN(C(=O)CSc2ccc(Cl)s2)CC1O N(C1CCc2ccc(Cl)cc21)C(C1C(NC(c2csc(C)c2C)=O)CCC1)=O C1(NC(c2c(C)nccc2)=O)CC2(CCN(C(=O)CCC3CC3)CC2)C1 C12(CNC(c3cn(CCC)nc3)=O)CCCCC1N(C(=O)CC(C)OC)CC2 N1(C(COCC)=O)CCCCC1CCN(C(=O)CCCC1CC1)C(C)C C1(NC(c2c(CC)cno2)=O)CC2CC(NC(c3cccnc3OC)=O)CC2C1 N1(C(C2(CC#C)CCC2)=O)C2CCC1C(NC(c1ccccc1SCC=C)=O)C2 C1(C(=O)NCC(CN(C(c2cc(COC)on2)=O)C)C)OCCOC12CCC2 c1(OC)ccc(C(=O)NCCC(C)NC(=O)Cc2ccc(C)o2)cc1[N+](=O)[O-] N(C1CCc2sc(Br)cc21)C(c1n(CC)nnn1)c1nncn1C N(C(=NCCCCl)NC1CC(C)(F)C1)C1CC(C(=O)OCC)C1 n1(C(C)C(=O)NC2CCN(C(C3(C)CC3(F)Cl)=O)C2C)cnc2ccccc12 C=C(C)CC(C(=O)NC(C(=O)OC)C1CC1)NC(C1CC1CCOC)=O N1(C(C(CC)OC)=O)CC2(CCN(C(c3[nH]ccc3-c3ccccc3)=O)C2)C1 C1(C(=O)OC)CN(C(c2nc(CNC(=O)C(C(C)C)SC)oc2C)=O)CCN1C C1(COC)(NC(=O)Cn2ccc(C)n2)CCCN(C(C2CCC(C)(O)CC2)=O)C1 C1(NC(Cc2n(C)ncc2Cl)=O)CC(F)CN(C(C2(C(F)F)CCCO2)=O)C1 N1(C(c2n(C(C)C)ccc2)=O)CCC(O)(CNC(C23CC(CC(C)O2)C3)=O)CC1 C1(C(N2CCN(C3CCN(C(CS(N)(=O)=O)=O)C3)CC2)=O)CCc2nncn2C1 c1(C(CNC(C(=C)CO)=O)C)ccc(S(C)(=O)=O)cc1 c1(C(=O)NCC2CCCCN2C(=O)CC2CC3CCC2C3)cncc(F)c1Cl c1(C(C)Oc2ccccc2)cccc(CNCc2cn(C)nc2-c2cccs2)c1 CC(C)CC(C1CCC1)NC(c1nnnn1C)(C1CCCCC1)C c1(C(N2C(CNC(C(CCN(C)C)O)=O)CCCC2)=O)c(Cl)nn(C)c1Cl C12(CCNC(C3(OC)CC3)=O)CCC1CN(C(c1ccnn1C(F)F)=O)C2 c1(C(=O)NCCOC2CCN(C(C=CCC)=O)C2)cnc(OC)nc1 C1(NC(COCc2n(C)ncc2)=O)CC2(C1)CC2N=c1nc(CC2CC2)[nH]s1 CC(CC(=O)NC1CCC(C(=O)NCCc2cn[nH]c2)C1)CC(C)(C)C N1(C(CNS(CC)(=O)=O)=O)CCCC(NC(=O)CCCn2cccn2)C1C CN1CCS(=O)(=O)CC1CC(=O)NCC1CC2(CO1)CC(=O)C2 c1(NCCN2CCC(OC)CC2)[nH]c(=NCCC2CC2C)nc2ncn(C)c12 C1(NC(C2ON=C(C)C2)=O)CN(C(=O)C=C2CN3CCC2CC3)CC(C)(C)C1 n1(CC(=O)NCCOCCNC(CCCOCC=C)=O)ncc(Br)c1C C1(NC(=O)CCC2CCCN2C(=O)C(Cl)Cl)(CO)CCCCC1 C1(c2cn(C(c3ncccc3Br)C)nn2)(C(=O)OC)CNC(=O)C1 N1(C(c2cc(CC)c(CC)o2)=O)CC(F)(F)CC1(C)CNC(c1csnc1C)=O Cc1cc(F)ccc1-n1cc(NC(=O)C(C(C)(C)O)Oc2ccccc2)nn1 C1(C)(C)CC(=O)NC(C)c2cn1nn2.N(C)CC.C(C1CC1)C1CC1 c1(-c2nc(NC(c3c(C)n(C4CCOC4)nn3)=O)sc2)ccc2c(C)[nH]nc2c1 C#CC1CN(C(C2CCC(C(F)(F)F)O2)C(=O)NC2CCOCC2)CCN1C CN1CCOC(C(=O)N(C)CC2CCCN2C(c2cccc(Cl)c2)=O)C1=O C#Cc1cc(C(=O)NC(CNC(=O)C(C)(C)OCCC)CC(F)(F)F)ccc1C c1(C(N2CCC(NC(C3C(C)C3C)=O)CC2)=O)cc(N(C)C)ccc1Br c1(CN2CCC(F)(C(=O)Nc3cnn(C4CC4)c3)C2)cc(Cl)c(Cl)c(Cl)c1 CC1CC(CC(=O)NCC2CCCC2)CN1C(=O)CN(C)CCOCCO C1(CC(N2CC(C)C(CNC(c3cn(CCF)nn3)=O)C2)=O)CC2CCC1CC2 O=S(=O)(c1cncc(Br)c1)N1CC2CC(C1)N2c1nccc(-c2ccccc2)n1 Cc1ccc(-n2cc(CONC(=O)CC3CCC(=O)N3C)nn2)cc1 Cc1cc(CNC2CCN(C(=O)C3CC3)CC2O)c(C)c(C)c1 C1(NC(c2c(C)ncnc2)=O)CC(C2CCN(C(=O)CCCc3ccsc3)C2)C1 C1(NC(c2ccc(CC)cn2)=O)CCC(C)N(C(c2cc(=N)[nH]cc2Br)=O)C1 C1(O)(CN(C(CCSC)=O)C)CCCN(C(=O)C(C)C(=O)N2CCOCC2)C1 CCC(C)C(C(=O)NC(C)Cc1cc(C)[nH]n1)NC(c1ccc([N+](=O)[O-])o1)=O N1(C(c2c(C)cccc2)=O)CC2CC(C(=O)NCC(O)CCC3CC3)C(C2)C1 C1(NC(CCN(C)CCO)=O)CCC(NC(=O)C(F)(F)C2CC2)C1 c1(OC)cccc2c1OCC2NC(=O)C(N1CCSCC(CO)C1)=O C1(NC(Cc2scc(C)c2)=O)CC2CN(C(=O)C(F)(F)C3(O)CCCC3)CC12 Cc1ncsc1C(=O)NC1COCC1NC(c1conc1C1CCC1)=O N1(C(c2cc(CCC)[nH]n2)=O)CC2(C(=O)NC(C)C(O)C(F)F)CC1CO2 c1(-c2nc(C3(C4CCC(=O)N4)CC3)on2)cc2c(Br)cccc2[nH]1 N1(C(C(F)=CCC)=O)CCC2CN(C(c3cc4c(Cl)cncc4s3)=O)CC2C1 C1(C(N2CC(CCCC)N(C(=O)CS(C)(=O)=O)CC2)=O)CC1C1(C)CCOCC1 CC1=NOC(C)(C(=O)NCC2CCC2NC(=O)COC2CCCCCC2)C1 n1(CC(=O)C2CC2)cc(CNC(=O)C(O)C2CC2)nn1.C1(CC)(CSC)CC1 c1(C(C)C)ccc(C(N2CC(CNC(=O)C(CN(C)C)N(C)C)C(C)C2)=O)cn1 C1(C(=O)NC(C(=O)OC)Cc2csc3ccccc23)CC2(CCC2)CCN1 c1(N2CCC3(C(C(N4CCC(CCOC)CC4)=O)C3)C2)nc(C)nc2c1CCC2 C1(CNC(C(C)Cn2cccn2)=O)CC12CCN(C(c1cnns1)=O)CC2 c1(C(N2CC3(CC(NC(C4(C#C)CCC4)=O)C3)C2)=O)cc2cccnc2o1 c1(OCC(=O)NCc2cccc(SC)c2)cccc(C#N)c1 c1(NC(c2nc(-c3ccc(Cl)cc3)ns2)=O)nnc2n1CCCC2 N1(CCCCC)CCC2CC(C(=O)N(CCO)Cc3cccs3)C2C1 N#Cc1ccc(C(N2CCN(C(=O)CC3COC4CC3C4)C3CC23)=O)cc1 c1(NCCc2cn[nH]c2)ccc2c(c1)CC2.C12CC1NC(=O)NC2C N1(C(C2C(CNC(c3c(C)cc(C)o3)=O)C2)=O)CC(=O)N(C)C(C)C1 c1(CC)sccc1C(N1CC(O)(C(C)NC(=O)C(C)NS(C)(=O)=O)C1)=O CC(C)(C)CC(C(=O)N1CCC(C2CC2)C1)NC(C1CCCC1)=O N1(C(CCCCNC(C)=O)=O)CCCN(C(c2ccc(C(N)=O)nc2)=O)CC1C C1(C(F)(F)F)(OC)CC(C(=O)N(C)CCNC(=O)CC2CCC(=O)N2)C1 c1(C(=O)NCC2C(NC(CCc3cc(OC)no3)=O)C2)cccc(N)c1C Cc1nc(CC(C)C)sc1C(=O)NCC1CCC1NC(=O)C(O)C(F)F c1(OC)ccc(Br)cc1C(CO)NC(=O)CC1(Sc2ccccc2)CCC1 c1(CC)onc(C2CCOCC2)c1C(=O)NCCc1ccccc1N C1(C(N2CC(CCNC(c3cc(O)cs3)=O)C2)=O)(OC)CCOCC1 C12(CNC(c3ccc(CC)cc3)=O)CCC1CCN2C(C1CC(S(C)(=O)=O)C1)=O Cn1c(C(=O)NC2(CO)CN(C(=O)Cn3cc(Br)c(=N)[nH]3)C2)nnc1S c1(OC)ccc(F)cc1C(N1CC(OCCNC(=O)CC(C)C(F)F)C1)=O C1(N(C(C2C(Cl)(C(=O)OC)C2)=O)C)CCC(NC(c2ccnnc2S)=O)CC1 C1(C(=O)NCC2CCSCC2)(NC(=O)C(C2CCCCC2)O)CCCCC1 C#CCCCCC(=O)NC1CC=C(C(=O)NC2(CO)CCCCC2C)C1 C1(CNC(C(CCC)NC(N)=O)=O)CC2(CCC2)CN1C(=O)CC1COC(=O)C1 C1(C(=O)O)(NC(=O)NC2COCC2n2cc(Br)cn2)CCN(C(C)(C)C)C1 C1(NC(c2n(CCC)ccc2)=O)CCC2CN(C(c3ccc(C)nc3)=O)CC2C1 c1(C(=O)NC(CCOC)CNC(=O)CCNC(=O)CC(C)C)ccc(O)cc1F C(c1ncccc1C)=CC(=O)NC(CNC(c1c(SCC)cncc1)=O)CO c1(C(=O)NCC(C(C(C)C)C)NC(=O)CCCN=[N+]=[N-])cnn2c(Cl)cccc12 CCC(O)C(C)C(=O)N(C)CC1(CNC(c2cn(-c3ccccc3)nn2)=O)CC1 C1(C(N2CCC(F)(C(N)=O)C2)=O)CC2(CC2)CN1C(=O)Cc1ccccc1F c1(C(N2C(CN(C(CCSC(C)C)=O)C3CC3)CCC2)=O)cccn2nccc12 c1(C(=O)NC(C(C(C)C)NC(c2n(COC)ncc2)=O)C)cc2cccnc2s1 CC1CN(C(C2(F)CCOC2)=O)CC(C)N(C(=O)C(=O)Nc2ncc[nH]2)C1 c1(NC(CCC)(c2nnnn2CCCF)C2CCCC2)ccc(CC)c(O)c1 C#CCC(CC#C)C(=O)NC(C)(CNC(=O)Cn1c([N+](=O)[O-])cnc1C)C(C)C c1(CC(=O)NCC2C(NC(CCSCC)=O)CCCC2)c(C)nc(O)nc1C C(=O)(C1=CC2C=CC(C1)C2)NC(C1(C(=O)NC2CCC2)CC1)C.COC N1(C(Cc2c(C)scc2)=O)CCC2CCN(C(c3ccc4cccnn34)=O)CC12 N1(C(=O)CCC2CC2)CCN(C(c2ccc(Br)c(O)c2)=O)C(CF)C1 c1(C(N2CCC(n3cncn3)C2)C(=O)NC2CCOC2)cc2n(n1)CCCO2 c1(OC)ccc(C(CNC(c2nc(Cl)oc2C)=O)NC(c2nnn(C)n2)=O)cc1 Cc1cc(C(N2CC(F)(F)CC2(C)CNC(c2cnccn2)=O)=O)c(F)cc1Cl c1(CC)nocc1C(=O)N(CCN(C(=O)C(C)n1cnnn1)C)C(C)C c1(C(C)=O)c(Cl)nc[nH]c1=NCCN(C(=O)C(C)(C)c1cncnc1)C(C)C N1(C(Cc2n[nH]c(=NC)s2)=O)CC(NC(c2cc(Cl)ccc2Cl)=O)C2(CC2)C1 N1(C(CN(CCC#C)C)=O)C(CC(N2CCC3CCC23)=O)C2CCCC12 C1(C(=O)NC(CC)C(=O)OC)CC(C)(C)CN1C(C1CC(=O)CC(=O)N1)=O C1(CC)CN(C(=O)CSC(F)F)CCC1NC(=O)CCc1cn(C)nn1 c1(C(N(C2CCC(NC(C(n3c(C)ncc3)C)=O)CC2)C)=O)cc([N+](=O)[O-])c[nH]1 c1(NC(C(C)Nc2ccccc2C(F)(F)F)=O)nccc2occc12 c1(CC)ccccc1C(=O)NCC1CCCC1N(C)CCOC C(=O)(C1=CC2CCC=CCCC12)N1CC(C)C(NC(c2cc(O)cs2)=O)CC1 c1(CNC(C=CCC)=O)cncc(NCCO)n1 Cc1cc(C(C)C(=O)NCC=CCNC(C2CCCN2C2CCOCC2)=O)c(C)o1 C1(CNC(c2c(CC)nc[nH]2)=O)CCC(C)N(C(c2nc(C3CC3)cs2)=O)C1 C1(c2cc(CC)c(C)cc2)CCN(N2CCN(C(=O)CSC)CC2)C1 C1(CCN2CC(NC(C(F)=CC)=O)C2)C(=O)OCC1(C)C c1(C(N2C(CCCNC(CCSC)=O)CCC2)=O)cc2ccncc2cc1F N1(C(CC=C)=O)CCCCC(NC(C2CN(C)CCO2)=O)C1 c1(SC)c(NC(c2cccc(C(C)=O)c2)=O)cnn1C N1(c2cc(NCc3ccc(CN(C)C)cc3)nc(C)n2)CCCCCCCCC1 Cc1ccc(CC(=O)NCC2CN(C(c3cc(CC(C)C)on3)=O)CCO2)cn1 C=C(C)CCCC(=O)N(C)CC1CCCC(NC(c2cc(C)n(C)c2)=O)C1 c1(C(N2CC3(C(NC(=O)CCc4cc(Cl)no4)CC3)C2)=O)csc2ccccc12 C1(C(=O)NCC(O)C2CCC2)CN(C(c2c[nH]c(=S)cn2)=O)CC(F)(F)C1 c1(CC)onc(C(=O)NCC(O)CC(=O)NCC(C)(O)C(F)F)c1C N1(C(CSC(C)C)=O)CC(O)(CNC(C2CCN(C(C)=O)C2)=O)C1 CC1CCC(C(N2CC(CO)C(CO)C2)=O)CN1C(c1nc[nH]n1)=O N1(C(CNC(=O)OC)=O)CCc2c(Cl)cccc2C1.C12CC(F)CN(C1)C2=O N1(C(CCCSC)=O)CC2CCC(CNC(c3c(C)nn(C)c3C)=O)C2C1 N1(C(C(C2(CO)CC2)NC(C2C(C)C2C)=O)=O)CCC(C)(CCO)CC1 n1(C(C)C)cnc(C(=O)NCCNC(=O)CCCc2ccsc2)c1 c1(C(=O)NC(C)C(=O)NCC2(C)CC2(C)C)cc2cnccc2[nH]1 CCC(CC)CC(F)C(=O)NCc1cc(C(=O)N(C(C)CS(C)=O)C)cs1 n1(CC=C)cc(C(N2CCC(C(C)NC(c3csc(C(F)F)c3)=O)C2)=O)cn1 c1(OC)cc(C)cc(C(=O)NCC(C2CC2)NC(=O)C(O)C2CC2)c1N CCCN=c1[nH]c(=NC)[nH]c(=NCC(C2CCCC2)N(C)C)[nH]1 Cc1nn(CC(C)C)c(Cl)c1C(N1CCC(O)(CCNC(=O)C(F)C2CC2)C1)=O Cc1cnc(C(N2CC(CC(=O)NCC3C(C)(C)C3(F)F)C3(CC3)C2)=O)c(C)c1 C1(C#N)(C(N2CC(C(C(=O)NCc3cc(COC)no3)O)C2)=O)CCCCC1 c1(C(=O)NCC2CCCC(CNC(C(COC)(F)F)=O)C2)cc(OC)cc(C)n1 C(=O)(C(CN(C)C)C(C)C)NCCN(CCC)C(C1CCSC1)=O C1(OCC)CC2CN(C(=O)CCC3(C)CC3(F)F)Cc3cccnc3N2C1 c1(C(=O)OC)cc(NC(C2(O)CCN(C(=O)C(C)NC(C)=O)C2)=O)ccn1 C(=O)(C(CC(C)C)n1ccnc1)N1CCC(NC(CCOCCCOC)=O)C1C c1(NC(C2N(C(c3cc(CC)[nH]n3)=O)CC(O)C2)=O)cnc(Br)c(Cl)c1 C1(NC(c2ccn(CCC)n2)=O)(COC)CCCN(C(=O)CCC(C)(C)OC)C1 N1(C(C2CCN(CC)C2)=O)CC(N=[N+]=[N-])CC1C(=O)N(C)Cc1cnc(C)cn1 Cc1[nH]nc(C(=O)NCCC2(C)CCN(C(=O)Cn3cc(C4CC4)nn3)C2)c1Cl C1(C(=O)NCC(CNC(c2c(C)cn(C)n2)=O)F)CCC(C)(C)CO1 C(=O)(C1c2c[nH]nc2CCC1C)Nc1nccs1.N12CCCC(C1)C(=O)NCC2C N1(C(C(C)C2CCCC2)=O)CCOC(CCNC(c2ncoc2Br)=O)C1 C(C(CO)(CO)NC(c1nccnc1N)=O)N(C(c1nc(OCC)oc1)=O)C CC1CN(C(c2ccc(Cl)cn2)=O)CCC1NC(C1CCOCC1)=O Cn1cc(C=Cc2nc(C3(O)CCOC3)no2)c(=O)n(C)c1=O CC1CN(C(=O)CCS(C)(=O)=O)CCN1C(C1C2COCC12)=O c1(SCC)ccccc1CC(=O)NC12CC(NC(=O)CCc3ccccn3)(C1)C2 c1(CC(=O)NCC(C)CN(C(=O)C(F)n2cccn2)C)ccsc1Br Cc1nn(C)c(C)c1CCn1c(N2CCC(C)(F)C2)nnc1C1CCC(=O)N1 Cc1c(C(=O)N(C2CC(NC(c3nccnc3N)=O)C2)C)cnn1C C#CC1(C(=O)N(CC)CC2CC2)CCN(C(c2ccc([N+](=O)[O-])[nH]2)=O)C1 N1(C(C(C)OC)=O)CCc2nc[nH]c2C12CCN(C(=O)C(C#N)=CC(C)C)C2 C1(CC#C)(C(=O)N(C)CCNC(C2CC2(c2cccc(Cl)c2)C)=O)CCCCC1 C1(N(C(C(N2CC(C(=O)OC)C(N(C)C)C2)=O)=O)C)Cc2ccccc2C1OC c1(OCC=C)ccc(C(=O)NC2COCC2CNC(C2CC2(F)F)=O)cc1 CC(C)C(O)C(C)C(=O)N(CC(C)(C)C(N1CCCN(C)CC1C)=O)C N1(C(C(=O)NCCS(=O)(=O)N(C)C2CC2)=O)CCCC(c2ccc(O)cc2)C1 C1(NC(c2cccc(-c3nc[nH]n3)c2)=O)CCCCN(C(=O)Cc2nccs2)C1 Cc1ccc(C2(NC(C)Cc3cnccn3)CCC2)c(C)c1 C(c1ccc(F)cc1)=CC(N1CC2(C1)CN(C(C1CC(CN(C)C)C1)=O)C2)=O c1(C(N(C2CCN(C(=O)CCCCc3cnc[nH]3)C2)CC)=O)ccc(F)c(C)c1 C1(C(=O)NC2(CCC(=O)NCC3(C)ON=C(C)C3)CCC2)CCC2(CCC2)C1 c1(OC)ccc(C(N2CC(NC(C3CCC4CC34)=O)CC(C)(C)C2)=O)c(O)c1F C1(NC(=O)CC2CC(F)(F)C2)CCCN(C(C2(CF)CC(F)(F)C2)=O)C1 Cc1ccc(Br)c(CN2CCC3(CC3C(=O)NCCC(C)(C)CO)C2)c1 c1(C(=O)NCCCCC(C)NC(C(CC)OC)=O)c(C(F)F)nc2n1CCCC2 c1(SCCOC2CCN(C(C=CCC)=O)C2)ccc2ccccc2c1.OC O=C1COc2c(NC(C3(c4nc5ccccc5s4)CCC3)=O)cccc2N1 Cc1sc(O)nc1C(N1CCC(C)C1CNC(c1cn(C)c(C(F)F)n1)=O)=O N1(C(C2(CC(C)C)CCNC2=O)=O)CCC(NC(=O)C=Cc2ccco2)C(O)C1 CC1(C)C2CCC(C2)C1(C)C(=O)NC1CN(C(=O)CCc2ncc[nH]2)C1 n1(CCC)cc(Cl)c(C(=O)NCC(C)CN(c2ncc(C(F)F)cn2)C)n1 C1(O)(CNC(c2scnc2Cl)=O)CCN(C(C2(CCF)CC2)=O)CC1 N1(C(CNC(CC)=O)=O)CCC2(CC2NC(=O)CC2CCCC(C)(C)O2)C1 C1(CNC(CCC=CCC=C)=O)CC2CCC1N2C(=O)C(C)(C)SC CCCCC(CNC(c1ccc(C(O)CF)cc1)=O)NC(c1occc1C)=O C1(NC(c2ccc(Cl)c(F)c2)=O)CCN(C(=O)CCc2cccc(O)c2)CC1F N1(C(COCC(C)C)=O)CCN(C(=O)C2=CCCOCC2)C(CC(C)(C)C)C1 C1(C(=O)NCc2ncccc2F)CCN(C(C2CC2(F)Cl)=O)CC1O N1(C(c2cc(OC)n[nH]2)=O)CCCC(C(C)NC(=O)C=CC(C)=O)C1 c1(OC)cc(OC)c(C(N2CCC(c3ccc(C)cc3)CC2)=O)cn1 N1(C(C2CC(C)OC2C)=O)CCn2ncc(CC(=O)N(C)C)c2C1 C1(O)(C(N(CCNC(c2c[nH]cc2C2CC2)=O)C2CC2)=O)CCOC1 c1(SC)ccc(OCC(=O)N(C)CC2CN(C(=O)CSC(C)C)CCO2)cc1 C1(C(=O)NCC2C(C)CCN2C(=O)CCCC2(C)N=N2)Cc2ccccc2C1 N1(C(CC(n2ccc(C)n2)C)=O)CCCC(C2CC2NC(c2ccc(C)s2)=O)C1 c1(C(N2CCC(NC(C(C)CC3CC3)=O)C2C)=O)cc2ccncc2cc1F c1(C(=O)NCC23CC(NC(c4c(C)nns4)=O)(C2)C3)c(C(F)(F)F)cncc1F Nc1ccc(C(=O)NCC(O)CNC(=O)CNC(=O)CC(F)(F)F)nc1F N1(C(CC2(C)OCCO2)=O)CCC(C)(C)C(NC(c2nc3ncccn3n2)=O)C1 Cc1nc(C(C)C)ncc1C(=O)NC12CCCC(NC(=O)C(C#N)C3CC3)(C1)C2 C(=O)(CCCC(C)NC(C1CCN(C)C1=O)=O)N1CCC(C(=O)OC)C1C c1(C(N2CCN(C(c3c(C)cc(O)nc3)=O)CC2C)=O)cccc(C#CCO)c1 c1(C(N(CC(CC)(C)C)C)=O)cc(C)n(CC)c1C CCCC(C)(C(=O)O)NC(=O)Nc1ccnc(NC(=O)OC(C)(C)C)n1 Cc1cc(Br)cc(C)c1CN1CCCC(CCNC(C2(O)CC2)=O)C1 c1(NCC2CCC(NC(c3cn(COC)nn3)=O)C2)ncc2c(n1)CCCCC2 C1(C(=O)NCC2N(C(c3c(OC)ccc(C)c3)=O)CC2)CN2CCN1CC2C C#Cc1cc(C(N2CCC(NC(C3CCS(=O)CC3)=O)C(CO)C2)=O)ccc1Cl C(=O)(CCC(C(C)C)NC(C1CCCC(=O)C1)=O)NC(COC)C1CC1 c1(C(=O)NC2C(NC(C(C(C)C)F)=O)COCC2)nn(C)c2c1CCCC2 O=C(CC=C(Cl)Cl)NC(c1cccnc1)C(=O)NCC1CCCCS1 C1(CC=C)(C(=O)O)CN(N2CC=CCC3(CCOCC3)C2)C1 CC(F)(F)CCCC(=O)N1CC2CC1C2NC(c1cnc(O)n(C2CC2)c1=O)=O S(=O)(=O)(c1ccc(C(N2CCCN(C(=O)C(C)(C)CO)CC2CO)=O)o1)NCC CC(C)C(C)C(CNC(c1cccnn1)=O)NC(c1cc(O)nc(C2CC2)n1)=O CC(CCNC(c1cnc(Cl)cn1)=O)N=c1cc(Cl)nc(C2CCCO2)[nH]1 CC1CN(C(c2c(CNC(=O)Cn3cnnn3)nnn2C)=O)C2(CC2)C(=O)N1 N1(C(COCC#C)=O)CCN(C(c2nnsc2C)=O)CC1CCC C(=O)(CC1=CCCCC1)NCC1CCN(C(C(CC)C(C)O)=O)C12CC2 C#CC1CCCCN1C(C)=O.n1(CC(=O)NCC2C(=O)N2)nc(C)oc1=O C12(C(N3CCOC(CC(=O)Nc4c(C)ocn4)C3)=O)CC1COC2(C)C C1(C(N(CCN(C(c2cnc(CC)nc2)=O)CC)CC)=O)Cc2nccn2C1 C(=O)(NN1CCCC1C(=O)NCC#CCCO)c1cc(CC)[nH]n1 C(=O)(C(O)C(C)(C)C)N1CCC(C)(C(=O)Nc2ccc(C(=O)OC)cc2)C1 N1(C(CCNC(=O)OCC)=O)CCCC1C1CCN(C(C2(C)CC2C)=O)C1 Cn1cnc2cccc(C(=O)NC3CCC(NC(=O)Cc4ccno4)C3)c12 Cc1ccc(Oc2cccc(CNC(=O)NC(C)C(C)CO)c2)cc1 c1(NC(CCCC)CCC)nccc(=NCCOc2ccc3c(c2)CCC3)[nH]1 N1(C(COCCOCC)=O)CCCCC1CNC(c1coc(CC2CC2)c1)=O N1(C(C(Cc2cn[nH]c2)NC(C2C(C(=O)OC)C2)=O)=O)CCC(F)(F)C(O)C1 c1(CC)nc(-n2cccc2)sc1C(=O)NCCCNC(C12CCC(CO1)C2)=O C12(NC(C3=C(C)CCOC3)=O)CCCC1(F)CN(C(c1ccccn1)=O)C2 c1(C(=O)N)c(F)cncc1Cl.Cc1nn(C2CC2)cc1C(=O)NCC1CC1C C1(CNC(C(C2(O)CCC2)NC(c2cn(CC)nn2)=O)=O)C(C)(C)C1(F)F Cc1noc(C)c1CN1CC(CCNC(=O)Cc2nc(C3CC3)cs2)C1 C(=O)(C(C)(C)CCS(C)(=O)=O)N1CC(NC(C(C)Sc2ccc(F)cc2)=O)C(O)C1 N1(C(C2CCC(CNC(c3cnn(CCO)c3)=O)C2)=O)CC2(CCOC2=O)C1 C(=O)(CC(C)C(C)(C)C)N1C(C)CC(c2ccccc2)C1.c12cn(nn1)CC2 n1(CC)ncc(C(=O)NC2CCC(C)(CNC(c3ccoc3Cl)=O)C2)c1C1CC1 C#Cc1cnc(NC2CC(CCNC(=O)C=CSC)C2)nc1 CC1CCC(Cl)=C(C(=O)NC2CCN(C(C3COC3)=O)CC2F)C1 c1(C(N2CC3(CN(c4nc(C)c(Br)cn4)C3)C2)=O)n[nH]c2c1CC(C)CC2 CC(C)(F)C(C)(F)CNC(C12CC(NC(C3CCCC3C(F)F)=O)(C1)C2)=O Cc1ccc(C)c(SCC(N2CCC(C(C)NC(=O)Cc3[nH]cnc3C)C2)=O)c1 c1(C(=O)NC(CC)C(=O)NCC(CNC(N)=O)(C)F)ccc(OC)nn1 c1(OC)cn(CC(=O)NC2CC2NC(C2CCCNC2=O)=O)c(C)cc1=O C(=O)(CC(C)(C)CN(C)C)N1CC(C)C(NC(c2cccc(NS(N)(=O)=O)n2)=O)C1 N1(C(C2(C)CC(F)C2)=O)CC2(C1)CN(C(c1ccc3ccnn3c1)=O)CCO2 CC(=O)CCCCCCC(=O)NC=O.c1cccc(C2CCN(C(c3ccccc3)=O)CC2)c1 C12(C(N3CC(C(=O)NC(CN(C)C)CCO)OCC3)=O)CC(C)(CCO1)C2 C(CS(=O)(=O)C(C)C)N(C(C1(N)C(C)CCC1)=O)C CC1CCCC(CC(=O)NC2(CNC(=O)CC3(O)CCCOC3)CCOCC2)C1 C12(NC(CC=C)=O)CC3CCC(C1C2)N3C(c1nc(O)sc1C)=O N1(C(c2cnn(C)c2Br)=O)CC2CN(C(=O)C#CC3CC3)CC2C1 CC(CCCCNC(C1(Cl)CC1(C)C)=O)NC(c1ccc(-n2cnnc2)cc1)=O c1(CSCC)cccnc1C(=O)NC1CN(C(=O)CCN2CCOC2=O)C2CC12 C(=O)(C#CC1CCOC1)N1CC(C(=O)Nc2cncc(C)c2)CC1(C)C CC(CCO)N=c1[nH]c2c(c(=NCC3(c4ccccc4)CC3(C)C)[nH]1)COCC2 c1(C(N2CCCC(C)(NC(C3CC=CCC3)=O)C2)=O)cc(F)cc(F)c1N N1(C(C(CC)CC)=O)CCC2CN(C(c3ccc(C#N)c(F)c3)=O)C(C)C12 CCC(CC(=O)NCC1(NC(=O)CNC(c2ccoc2)=O)CCOC1)C1CC1 c1(C(N2C(CC=C)(C(=O)NC3C=CCCC3)CCC2)=O)ccc(=O)n(C)n1 c1(C(=O)NCC(CNC(C2(F)CC2C)=O)OC)ccc(N)c(OCCO)c1 C1(NC(c2c(Cl)cn(C)n2)=O)CC2(CCCN(C(=O)CC3CCC(=O)CC3)C2)C1 c1(CN(C)Cc2cccc(OCc3cccnc3)c2)ccc(Br)cc1F C1(C(N2CCC(O)(Cn3cc(C(C4CC4)C4CC4)nn3)CC2)=O)CC2CCC(C1)S2 CCC(CO)CN=C(NCC1CC1(Cl)Cl)NC1CCN(C(=O)C(C)C)CC1 N1(C(c2cc(OC)nc(F)c2)=O)CC(NC(=O)CCNC(N)=O)CC12CCCC2 C(=O)(C(C(F)(F)F)C(F)(F)F)NCC(CCNC(=O)C(c1ccc(F)cc1)F)O Cc1nc(C(=O)NC2CC(C(=O)NCC3CC(=O)N(C4CC4)C3)C2)ccc1C#N CCC(CC)C(C(=O)NCC(C)(C1CC1)NC(=O)Cc1ccc(F)cc1)OC n1(CCC(N2C3C(NC(C4(C#C)CCC4)=O)CC(C3)C2)=O)ncc2ccccc12 n1(CC)nccc1C(N1CCC(CN(C(=O)C(C)c2ccco2)C)C1)=O C1(C(=O)NCC(CN(C(C)=O)C)C)Cc2cc(F)cc(F)c2O1 c1(C(=O)Nc2cccc(NC(c3c(NC)scn3)=O)c2)cccc(C2CC2)c1Cl N1(C(C2(C=C)CCOCC2)=O)CCN(C(=O)CC2CC(C)(C)CO2)CC(C)(C)C1 c1(C(=O)NCC(C(=O)NC2(CC=C)CCOC2)N(C)C)cccnc1C C1(C(=O)NC(C)Cc2ccc(C(F)(F)F)cc2)CCCNS1(=O)=O Cc1cc(C(=O)NC2CC(NC(=O)COCCCC(C)C)C2)co1 C1(CC=C)CCCCC1C(=O)NCC(N1CCC(N(C)C)C1)=O N1(C(C(CC=CCC)C)=O)CC(C(=O)NCC(N2CCCC2)C)C(F)(F)C1 N1(C(C2CC(=C)C2)=O)CC(NC(C23CC(c4ccccc4)C2C3)=O)CC(C)C1 c1(CC)ccc(C(=O)N(C)CC2(NC(=O)CS(=O)CC)CC2)c(C)c1 C(=O)(CC(C)CC(=O)NC(C)(C)C(C)CC(=O)N(C)CCn1ccnc1C)OC c1(C(=O)NCC2CCCC(NC(C3(C#C)CC3)=O)C2)c(CC)cccc1C C1(C(N2CC(OCC(C)C)C2)=O)(NC(=O)CN(C)C2CC2)CCN(C)C1 N1(C(C2C(C(C)C)C2)=O)CCC(OCCNC(=O)CSc2ccc(Cl)cc2)CC1 c1(N2CCN(C)C(C(F)(F)F)C2)nc(=NCC2CCOC2(C)C)[nH]c2cc[nH]c12 C1(C(N2CC(C#N)(F)C2)=O)CC(NC(=O)COCc2nc[nH]n2)C12CCC2 c1(C(=O)NCC2(CNC(C3CCOC3)=O)CC23CCC3)nnn2c1CSCC2 N1(C(c2cccc(Cl)c2Br)C(=O)NC)CCS(=N)(=O)C(C)C1 C1(CC(=O)NC(CCNC(CC2(CSC)CC2)=O)(C)C)CCCC1(F)F CC1CC=C(C(=O)NC(C(N2CCC(CO)C23CCC3)=O)C(C)(C)C)CC1 c1(OCCOCC)cc[nH]c(=NCCC(C)NC(c2c[nH]c3cccnc23)=O)n1 c1(C(=O)NC(CC#C)(C)C(=O)NCC2CCCCCCC2)cc2ncccc2[nH]1 Cc1ncc(C(=O)NC2(C)CN(C(=O)CNC(=O)CC3CCCC3)C2)cc1N Cn1cc2c(C(=O)NCC3CC3CNC(=O)Cc3cnc[nH]3)cc(F)cc2n1 c1(C(C2CC(NC(=O)C3=CCC3)C2)NC(C2C(OCC)C2C)=O)ccc(F)cc1 Cc1nc(O)nc(C)c1CC(N1CCC(CO)(NC(=O)CN2CCC(C)C2)C1)=O c1(C(N2CC3C(C2)N3C(C23CC(C2)C3)=O)=O)ccccc1CO C12(C(N(CCCC)CCCO)=O)CC(CN(C(C3CN4CCN3CC4)=O)C1)C2 C=CC1(C(N2CCC(O)C(O)C2)=O)CCN(C(c2cncs2)=O)C1 CCCC(CNC(=O)CC1CCC(=O)N1C)C(=O)N1CCC(C)(C#N)C1 CC1CCN(C(=NCCC2CCCC2)NCC(=O)Nc2cccs2)C1 N1(C(C2C(C)CCC2)=O)CCN(CCN2CCN(C(=O)C(C)(C)CO)CC2)CC1 C(=O)(C(CNC(C1C(=O)NN=C1C)=O)CC(C)C)NCC1CCN(CC)C1 n1(CC(=O)NC(C(C)NC(CC2CC(=C)C2)=O)C)cc(-c2ccccc2)cn1 n1(CC)cccc1C(N1CC(CC)(NC(c2cn(CC(=O)N(C)C)nn2)=O)C1)=O N1(C(CC#N)=O)CCCC(O)(CCNC(c2c(Cl)cccc2Cl)=O)C1 C1(C(C)C)CN(C(c2csnc2Cl)=O)CCCN1C(=O)C#CC(C)(C)C c1(-c2n(CC(=O)N(C)C)nc(C3CCCCCC3)n2)ccc2c(c1)OCO2 C1(NC(c2nnc(O)cc2O)=O)CC2CCC(C1)N2C(c1cccc(=S)n1O)=O c1(CC)ccc(C)cc1C(=O)NC1CC(O)CN(C(=O)C(=O)NC(C)C)C1 O=C(CC1=CCOCC1)NCCC1CCCN1C(=O)CC1CCCC1(F)F C1(NC(C2CCCS2(=O)=O)=O)CCC2CCN(C(c3cnc4n3CCS4)=O)C1C2 C1(CC)CC(C(=O)N(C)Cc2cncn2C)CCN1C(=O)Cc1cnc(C)s1 C1(CN(C)C)CCCC1C(N1CC(C)(NC(c2cc(C3(C)CC3)on2)=O)C1)=O CCC(C(=O)NC1C=CC(CC(=O)NCc2ncc[nH]2)C1)SC Cc1cc(C(N2CCC2CNC(c2cc(Cl)cs2)=O)=O)c(C)cn1 c1(CC)ccnc(C(=O)NCC2(CN(C)C(c3n[nH]c(C(C)(C)C)n3)=O)CC2)c1 N1(C(c2cc(C)cc(C)n2)=O)CCC2(C1)CN(C(c1csnn1)=O)CCO2 Cc1nnc2n1CC(C(=O)NC13CCC(CC1)N(C(=O)CN1CCCCC1)C3)C2 C1(C(=O)NCC(c2nccs2)C)(NC(=O)CCC2CC2)CC(F)C1 C1(C(=O)NC(C)CCNC(c2cccc([N+](=O)[O-])c2)=O)CCC2(CC1)CC2(F)F CONC(=O)C(=O)N1CCOC(C(C)NC(=O)COc2ccc(O)cc2)C1 C1(C(N2CCC2(C)CC(N2CCCC2CC2CCC2)=O)=O)OCC2CCCC12 C(=O)(C(C#N)C(C)C)NC1C=CC(CC(=O)NC(CCSC)C)C1 C(CC(C)C)(C(=O)NCCC(O)C1CC1)NC(c1ccc(NC)cn1)=O c1(C(=O)NCC2C(NC(CCCOCC)=O)CCC2)cnc(OC)nc1C N1(C(c2ccc(NC(C)=O)s2)=O)CCC2(CC2C(=O)NCC2CCN(C)CC2)C1 c1(C(C)(C)C)nnc2n1CC(C(=O)NCc1cncc(Cl)c1)CC2 C=CC1(CC(=O)NCC(c2ccccc2)NC(=O)C(C)CC2CC2)CCCCC1 c1(C(=O)NCC(O)C2(Cl)CC2)cc2cc(Br)cnc2o1 CCC1(C(=O)NCC(c2ccc3c(c2)OCCO3)O)CCCc2ccccc21 CC(C)(C(=O)N1CCN(C(=O)CC2CCC(F)(F)CO2)C(CF)C1)C(N)=O C1(CNC(c2cnccn2)=O)CCC2CN(C(C3CC4(C3)CC3(CC3)C4)=O)CC12 N1(C(CNC(=O)NC)=O)CCN(C(c2cc(NC)cnc2C)=O)C(C)CC1C C(CC(F)F)(C(=O)NCCCC(=O)NC)NC(C1ON=C(CC)C1)=O CC(C)C(Cn1ccnc1)N(CCC(F)(F)Cl)C(=O)CCNC.C(CCBr)O C1(CNC(CCCOCC)=O)C2CCCC1N(C(c1sccc1OC)=O)C2 C1(NC(=O)CCSc2cccc(F)c2)CN(C(=O)C2=CCOC2)CC2CCCC12 C1(C(=O)NC2CCN(C(C)(C)C)C2)CCCC(C(=O)Nc2ncccn2)CC1 C1(C(=O)NC(C2CCCCC2)CNC(=O)C(F)=CC2CC2)CC2CCC1O2 C1(C(=O)NCC2CCCC(CNC(C3C4CCCC34)=O)C2)CCn2cncc2C1 c1(C(N2CCC(C(C)NC(C3CC(OC)C3)=O)C2)=O)cc(Cl)cc(Cl)c1 c1(NC(C2CSCCN2C(=O)CO)=O)cncc(Cl)c1Br Cc1nc2cccc(C(=O)NNC(=O)C3CCC(=O)N3)n2n1 c1(SCC(=O)NCCCNC(CCc2cc(C)sc2C)=O)ncnc2[nH]cnc12 N1(C(C(C)SCC)=O)CC2(CCN(C(=O)COc3c(C)occc3=O)CC2)C1 CC1CN(C(=O)COC(C)(C)C)CCC1NC(=O)C(C)(C)Br C1(C(N(CC(CC)NC(c2cn(CCCF)nn2)=O)CC)=O)CCS(=O)(=O)N1C CC1(CO)CCCN1C(c1ccc(CNC(c2cnns2)=O)cn1)=O Cc1cc(F)cc(C(=O)NCC2CN(C)CCN2C(=O)COC2CCOC2)c1N N1(c2nnc(C(C(C)(C)C)O)n2Cc2cccs2)CCOCC2(CCOCC2)C1 C1(CC(=O)NC2(C(=O)NC3(CSC)CC3)CC2C)CCCC2CC12 Cc1noc2nc(C3CC3)cc(C(=O)NC(C)CNC(c3ccnnc3)=O)c12 Cc1nsc2ncc(C(N3CCCC(C)C3C(=O)O)=O)cc12 C1(c2nc(C(CC)CC)nn2-c2c(C)noc2C)CCC2(CCC2)O1 c1(C(=O)OCC)cc(C(=O)NC(CNC(C2CCC(C)C2)=O)C2CCC2)nn1C c1(-c2nc(C(=O)NCC(=O)N(C)Cc3ccc(Cl)cc3)sc2)ccc(Cl)c(Cl)c1 c1(C(=O)NCC(CC)(CC)NC(c2cccc(C)c2O)=O)ccc2nonc2c1 Cc1cc(C)c(C(N2CCC(C(C)(C)C)(CNC(=O)CN3CCOC3=O)C2)=O)s1 c1(NC(c2ccc(C)s2)=O)ccc(-c2cncc(F)c2)cc1 c1(COC(C)C)nc(-c2cncnc2)n(CC2CCCO2)n1 CN1CCCC1C=CC(=O)NCCNC(C1COCCN1C1CCCC1)=O CCS(=O)(=O)CC(=O)NC(C(=O)N(C(C)C(C)(C)O)C)C1CCC1 CC(C)(C)C1=NOC(CN=C(NC2CCOCC2)NC2CC2C(F)F)C1 C(=O)(C(Cc1cc[nH]n1)NC(c1cscc1OC)=O)NCCC(=O)OC CC(C)C(C(=O)NCC1CC(NC(=O)CCCNC(N)=O)CCO1)n1ccnc1 CS(C)(=O)=NC(=O)C(=O)N1CC(NC(c2cccc(C(F)(F)F)n2)=O)C(O)C1 N1(C(C2(CC)CCCN2C(c2cccnc2)=O)=O)CCCNC(=O)C1C N1(C(c2c(C)nsc2)=O)CCC2(CCOCC2)C(NC(c2nnc(S)n2C)=O)C1 Cn1cncc(C(N2CCCC(CNC(=O)Cc3ccoc3)C2)=O)c1=O n1(CC(C)C(=O)NC(CNC(c2cnccn2)=O)CO)ncc2c1CCCC2 c1(CCC(=O)O)nc(O)n[nH]1.c1(C(N(C2CC(OC)C2)C)=O)ccn(CCF)n1 C1(C(C)(C)C)(CNC(C(C)(C)OC(C)C)=O)CCN(C(C2CCCN2C=O)=O)C1 c1(Cc2occ(C(N(C(C(=O)OC)C)CCO)=O)n2)ccc(OCC)cc1 N1(C(CCc2onc(CC)n2)=O)CCC(CN=c2nn[nH]n2C)C(C)C1 Cc1ccc(Br)c(C(N2CC3C(C2)N3C(=O)C(C)Sc2ccccn2)=O)c1 C1(NC(c2cnn(C)c2N)=O)CC2CCC(C1)N2C(C1(C#N)CCOC1)=O N1(C(C(C)OCOC)=O)CCCC(C(C)NC(c2cc(C3CC3)no2)=O)C1 Cc1cc(N)cc(C(N2CCOC(CNC(=O)CC3CCCSC3)C2)=O)c1F c1(C(N2C(CNC(C(CCC)CC)=O)COCC2)=O)n[nH]c2cc(C)ccc12 C1(C(C)(C)C)(CNC(C2CCCS2(=O)=O)=O)CCN(C(=O)COCC(F)F)C1 C1(C(=O)NCC(CNC(=O)COC2CCCC2)F)C2CCC1(c1ccncc1)C2 C1(NC(C2CCC(F)(F)CC2)=O)CN(C(C23CCCC2C3)=O)Cc2ccnn2C1 C(C(C)(C)CCCO)NC(C(CSC)(C)NC(=O)C(O)C1CCC1)=O N1(C(C2CC(=O)NC2=O)C(=O)OCCNC(=O)OC(C)(C)C)CCCCCC1 c1(OC)ccc(-n2cc(-c3ccc(NCc4ccccc4)cc3)nn2)nn1 c1(OC)ccc(F)c(C(=O)NC2CC(CNC(c3ccc[nH]3)=O)C2(C)C)c1 c1(C(N2C(C)(C(=O)NCc3ccno3)CCC2)=O)c(F)c(F)c(O)c(F)c1F C(=O)(C1=CC2CCCC12)N1CC(CNC(c2nc(COCC)sc2)=O)(OC)C1 C1(C(=O)NC(C2CN(C(c3csnc3Cl)=O)CCO2)C)(N(C)C)CCOCC1 C(=O)(C(F)(CNC(C1CC2CC(=O)C1O2)=O)C(C)C)N(C)Cc1n(CC)ncc1 c1(C(N(CC(CC)NC(CSCCC)=O)C)=O)c(OC)cnc2ccccc12 C(=O)(C(C)(C)C(C)NC(=O)CCCCCF)N1C(COC)COCC1 c1(C(=O)NC2CC(C)(CNC(c3cc(OC)no3)=O)C2)ncccc1Br C=C1CC(C(=O)NCCCN(C(=O)CC2CCC2(C)C)CC)(C(F)F)C1 CC1CN(C(C23CCOC(C)(C2)C3)=O)CCN1C(=O)C(O)Cc1cn(C)cn1 C(=O)(C#CC1(C)CCCO1)NCC(c1ncc[nH]1)C c1(CC(=O)NCC2CC2NC(c2cc(CO)ccc2Cl)=O)cc(O)nnc1O C(=O)(C(C)(O)CC(F)F)NCC1(CCNC(C=COCC)=O)CC1 c1(C(=O)NC(CNC(CC(CC=C)(C)C)=O)C)oc(S(N)(=O)=O)cc1C CCC(C)C(O)CC(=O)NC1CC(C(N2CC(C)(C#N)C2)=O)C1(C)C CCC(CCCC(=O)N1CC(C2CC2)C1)NC(c1cnc(C)nc1C)=O N1(C(c2ccc(-c3nc[nH]n3)cc2)=O)CCN(C(c2ccns2)=O)C2CCC12 c1(C(=O)NC(CC=C)CNC(=O)C(F)Cc2ccccc2)ccnc2ccsc12 c1(C(N(CC(CC)NC(c2c(C)nsc2N)=O)CC)=O)cnc(N(C)C)nc1 c1(C(N(CC(CN(C(=O)CC2CSC2)C)O)C)=O)ccc(F)c2c1OCC2 N1(C(C2N(C)CSC2)=O)CCCC2(CCN(C(c3cnn(CC4CC4)c3)=O)C2)C1 N1(C(CC=CCNC(C2(C3CC3)CC(=O)C2)=O)=O)CCc2c(O)noc2C1 Cc1nc(NCC2CCCCO2)cc(N(C)Cc2csc(C3CC3)n2)n1 C(=O)(C1=CCCN(C(=O)C(O)c2ccsc2)C1)NCCC=CCCC C1(C(=O)NC2C3CN(C(C(C(C)C)NC(C)=O)=O)CC32)CCC(=O)N(C2CC2)C1 Cc1ccsc1Cc1nnc(N2CCCCC2)s1 C1(C(N(C)CC2CCCN2C(C2CC3CCCC23)=O)=O)CC(C(C)(C)C)=NO1 N1(C(CC2(C)CN(C(c3c(C)n[nH]c3C)=O)C2)=O)CCC(O)(CF)CC1 Cn1nc2ccc(Br)cc2c1S(=O)(=O)NNC(=O)c1ccco1 CCC(Cc1cccc(C)c1)C(=O)NC(CNC(C1(F)CCCCC1)=O)CO C#Cc1ccc(C(=O)NCC(C)(C)NC(C2CCSC2)=O)cc1F c1(C(c2n(CC)nnn2)NCCCC2CCOC2)c(I)ncn1C c1(C(=O)NC2C(CNC(=O)CC(C3CC3)C3CC3)CCC2)ncc(Br)cc1O C1(CN(C(=O)CSc2cccc(OC)c2)CC)CCCCN1C(=O)COC C1(NC(c2ncc(C)cc2C)=O)C2CC3CN(C(=O)CC4CCCN4C)C1C3C2 C(=O)(C(CC(N)=O)NC(c1cccc(F)c1)=O)NC(CCSC)C c1(C(N(CCCCCC(=O)NCCN(C)C(N)=O)C)=O)cccc2[nH]ncc12 c1(C(=O)NCC2CC(C(=O)NCc3cnc(C)o3)C2)ncn2ccccc12 c1(C(N(CCCN(C(COCCCC)=O)C)C)=O)cn(C)nc1-c1ccoc1 N1(C(c2ccc(CC)s2)=O)CC2CC(NC(c3c(C4CC4)noc3C)=O)C1C2 c1(OC)cc2[nH]ncc2cc1C(N1CCCC2(CCN2S(=O)(=O)C2CC2)C1)=O N1(C(C(C)n2ccnn2)=O)CCN(C(=O)C=Cc2cncn2C)CC1CCO c1(C(N2CCC(C)C(CNC(C3(CF)CC3(F)F)=O)C2)=O)cccc2ccsc12 C(=O)(N=c1cc(SC)n(C)[nH]1)C1CC2CN(C(CCC#CC)=O)CC1C2 C(C)(CCCCCO)NC(CC(COC)NC(C1CCCC(C)CC1)=O)=O c1(C(N(CCCCN(C(CC(CC)C)=O)C)C)=O)ccc(C(=O)OC)cc1OC CCC(CCC(=O)NCC(C)(C)C(C)(C)O)NC(c1ccnnc1)=O c1(C(N(CCNC(Cc2c(C)cc(O)cc2)=O)C(C)C)=O)n[nH]c2c1CCSC2 N1(C(C2C(C#N)C2)=O)CCN(C(=O)Cc2cnc[nH]2)C(CO)C1 CCCCCCCCCC(=O)N1CC(CC(C)NC(C2CCC3(CCC3)C2)=O)C1 c1(C(CC=CCNC(c2cc(C(C)C)on2)=O)=O)cc(Cl)cc(Cl)c1O n1(CC)cnc2c(N3CC(=O)NC(C)(C)C3)nc(=NCCC(F)F)[nH]c12 C=C(C)C(CC(=O)NCC(C)(CNC(c1cnc(C)[nH]c1=N)=O)OC)OCC c1(C(=O)NC2C(C(=O)NCc3cc(C)ns3)CC=CC2)c[n+]([O-])c(C)cn1 C1(CN(C(c2c(CC)scn2)=O)C)CC(F)CN1C(c1ccccc1C(C)O)=O c1(NC(C2N(Cc3ccc(OCCCC)cc3)CC2)=O)ccc(Cl)cc1C C(C(C)NC(N1CCC(c2ncc(Br)cn2)CC1)=O)(C(F)(F)F)OC CC1C(NC(C2CCOC2C(F)(F)F)=O)CCCN1C(=O)CSCCC#N c1(COCC)nc(C)c(C(=O)NC2CC2NC(c2cnn(CC)c2Br)=O)s1 O=C(CCCCCCNC(=O)C1=CCSC1)NCCCc1nc[nH]n1 Cc1cc2n(n1)CCCN2C(=O)NC(c1ccc(C#N)cc1)CF C1(NC(CCCCOCC)=O)CC(NC(c2ccc(SC3CC3)s2)=O)C12CCC2 C1(C(=O)NCc2c(CNC(c3c(C)nn[nH]3)=O)cccc2)CC2CCC1CC2 N1(C(c2c(NC)scn2)=O)CCC(C)(CNC(=O)CCC23CCC(CC2)C3)C1 n1(C(C)C)cccc1C(=O)NCC1CCN1C(=O)CCc1ccccn1 c1(SC2COC(C3(C#C)CC3)C2)nc(C2CN(C(=O)OC)C2)ccc1C#N C=Cn1nncc1C(=O)NCC1CC1C(=O)NCCN1CCCCC1=O N1(C(C(CCC=C)NC(C(CC=C)C)=O)=O)CCc2nc[nH]c2C1 N(C1CCCc2occc21)C(C(n1cc(C(c2ccccc2)OC)nn1)C)=O N1(C(C(CC(C)C)C)=O)CC2(CCCC2NC(c2cnc3sccn23)=O)C1 N1(C(c2cncs2)=O)CC2OCCN(C(c3cc4c(s3)CCC4)=O)C2C1 C1(Nc2nc(N(C3CC(OC)C3)C)c3c(n2)cc[nH]3)CC(=O)NC2CCCCC12 c1(OC)cccc2c1OCCCC2NC(=O)NC1COCCC1N=[N+]=[N-] c1(CC)ccc(C2(NCCCc3ccns3)CCC2)cc1 NS(=O)(=O)C1(C(N2CCC(F)C(NC(c3ccc(O)cc3)=O)C2)=O)CCCC1 c1(-c2cccc(NCc3c(N)nccc3)c2)ccc(Cl)c(Cl)c1 C1(CC(=O)NCCC2OCCN(C(C)=O)C2)CCCC(C)(C)C1 C(=O)(C1=CCC2CCC1N2C(c1c[nH]c(=S)cn1)=O)N1CC(C)CC(C(=O)OC)C1 C1(C(=O)NC(CC#C)CO)CCCCN(C(=O)CC2CCOC2=O)C1 n1(CC)cc(CCOC(c2cnn(C3CC3(F)F)c2)=O)cn1 c1(CC)cccc(F)c1C(=O)NC(COC)CNC(=O)C#CC(C)(C)C S(=O)(=O)(c1cnn(CCF)c1)NC(C(C)(C)C)c1ccccc1 N1(C(C2N(CC)CC2)=O)CC2(CCCN(C(C3(C)CCCN3C)=O)C2)C1 c1(C(C)=O)ccc(C(N2CCN(C3CN(C(=O)CC4C=CCC4)C3)CC2)=O)cc1 C(=O)(CCCCCF)N1CC(NC(C(C)OCC#C)=O)(CO)C1 c1(C(=O)NCC(CCNC(C(CC)(C)CO)=O)O)cccc2nc(O)ccc12 c1(CC)c(C(=O)NC2(C)CCN(C(C3(NC(C)C)CC3)=O)C2)[nH]c2ccccc12 N1(C(=O)CSC(F)F)CC2CC(C1)N(C(C1CC(F)(F)C1)=O)C2 O(NC(=O)C(C)(Cl)Cl)CC(=O)N(C1C(C)COCC1)C N1(C(C2CN(C)C(=O)C2)=O)CCC(O)(CNC(c2cc(O)cs2)=O)CC1 N(C)(C1CCc2cccc(Br)c21)C(C1CC(OC)CN1C(=O)OC(C)(C)C)=O CCS(=O)CC(=O)N(CCC(C(C)C)NC(=O)CC1CCCOCC1)C c1(C(=O)NC2CCN(C(c3ccc(CC)cn3)=O)C2(C)C)ccccc1[N+](=O)[O-] C#CC(C)(C)C(=O)N(C)CC1CCCN(C(C2CCC2(OC)OC)=O)C1 N1(C(CN2C(C)CCCC2)=O)CC(C2CN(C(=O)CC(C(F)F)n3ccnc3)C2)C1 N1(C(c2cnc(C)n2C)=O)CCC2C(NC(=O)C(C)C3CCCO3)C2C1 C(=O)(C1CCCc2ccccc21)Nc1ccc(-n2c(C#N)cnn2)cc1 N1(CCN2CC(C(C)C)C(N)C2)CCCC(CC2CCCCC2)CC1 C1(C(N2CC(O)(CN(C(=O)C3=C(Cl)CCOC3)C)C2)=O)CC2(C1)CC21CCC1 N1(C(c2cc(OC)n(C)n2)=O)CCN(C(c2ccoc2Br)=O)CC1C1CC1 C1(C)(C(=O)Nc2cccc(NC(C)=O)c2)CCCN(C(C2C=CC(=O)N=N2)=O)C1 C1(CC)CN(C(c2cnc(C)cn2)=O)CC1CNC(=O)C(C)Sc1nncn1C C1(CCNC(C2C=CCCC2)=O)CCCN(C(=O)CC23CC(C2)C3)C1 CC1CCN(C(=O)C(CCN(C)C)NC(C2CC3(C2)CC(O)C3)=O)C(C)C1 CCCCCCCCNC(C1CCCN(C(C2CCCN2C(=O)NC)=O)CC1)=O Cc1ccc(NCC2CCCCC2NC(=O)OC(C)(C)C)n2ncnc12 C=CCCCC(C(=O)NOC1CCOC1)NC(=O)C(C)C(F)F c1(OC)ncccc1C(=O)NCc1ccc(C(=O)NCCC(F)(F)F)nc1 N1(C(CC)=O)CCC(N(C(C2CC(=C(F)F)C2)=O)CC)CC1.N12CCC(C1)C2=O CCC(C)OCCCN(CC(=O)NCCN(C)C(C1CC1C(C)(C)C)=O)C c1(NC(=O)CC2COCCO2)cnc2c(c1)CN(Cc1ccc(O)cc1Br)CC2 C12(C(=O)NC(CNC(C3C(COC)C3)=O)C)CC3CC1C2C3(F)F CC(C)(CC(=O)NCC1CCC(C(N2CCOC(CN=[N+]=[N-])C2)=O)CC1)C1CC1 CC1CCCc2ncc(C(=O)N(CCCNC(c3nncs3)=O)C)n21 c1(C(c2n(CCOC)nnn2)NC2CCSC2)sc(C(=O)OC)cc1Br C1(NC(c2ccc(C(=O)OC)n2C)=O)CN(C(=O)C(O)C(F)F)C2(CCCC2)C1 c1(C(=O)NCCCOCCCNC(C2(SCC)CC2)=O)ocnc1C c1(COCCNC(C(C)N(C(CC2CC(=C)C2)=O)CCC)=O)ccccc1 Cc1ccc(OCC(=O)NCC(C)(C)CNC(C2(O)CCOCC2)=O)c(F)c1 c1(C(=O)NCC2(Cn3cc(-c4c(Cl)cn(C)n4)nn3)CC2)cncc2ccsc12 CC1CC(CNC(=O)COCCc2ccc(Cl)s2)CCN1C(C1CCC1)=O c1(OC)ccc(-c2nnn(CC(=O)NCc3nocc3C)n2)cc1OC(F)F C(=O)(C1=Cc2ccccc2C1)NC(CC)CNC(=O)CSc1ccccc1F C(=O)(C(CC(C)(C)C)NC(C1CCC(C)(C)OC1)=O)N(C)CC1(C#N)CC1 C1(CNC(C2CC(CCO)C2)=O)CC2(CO1)CN(C(=O)CC1CC1)C2 CCCCN=C(NC(C)CC)NCC(Cc1ccco1)CO c1(SC)cccc(C(N2CCC(O)C2)C(=O)NC2CCC2)c1.C1(C(C)C)C(=O)N1 C1(N(C(CC2CCN(C)C2)=O)C)CCN(C(=O)C2=NOCC2)CC12CC2 N1(C(C(C)SCC)=O)Cc2cccc(CNC(=O)C=C3CCC3)c2C1 Cc1cc2[nH]c(C(=O)NCC(C)(C3CC3)NC(=O)C#CC3CCC3)cc2s1 Cc1scc(C(=O)NC(C2CCCN2C(=O)CNC(=O)C2CC2)(C)C)c1C S(=O)(=O)(c1ccc(CCN)cc1)N1CCN(CC)C(=O)C1 c1(C(=O)NC2CN(C(c3cc(OCC)ncc3)=O)C(C)C2)ccc(C)c(N)c1 N1(C(CCCCOCCC=C)=O)CC2(CCC(NC(=O)CC(C)(C)SC)CC2)C1 CCCC(C)CNC(c1cnn(CCNC(c2ncoc2C)=O)c1)=O C1(CNC(CCCCCC#C)=O)CCCC12CCN(C(=O)CS(=O)CC)CC2 C1(NC(=O)C2=CS(=O)CCC2)CCC2(CCN(C(=O)CCOCC(F)F)CC2)C1 Cc1cnn2ccc(C(=O)NC3CN(C(c4cnn(C5CCC5)c4C)=O)C3)nc12 CCCCCC(F)C(=O)NC1CCOCC1NC(=O)C(c1ccc(C)cc1)F c1(C(N2CC(C(C(=O)NCCc3n(CC)cnn3)O)C2)=O)ccc([N+](=O)[O-])[nH]1 C1(NC(CCC2CCC(N)C2)=O)CC(C2CC2)C1 n1(CCN(C)C)cc(C(=O)NCC(C)(CO)NC(C2CCC2(F)F)=O)nn1 N1(C(c2cc(CCNC(c3n(CC)ccn3)=O)on2)=O)CCC(C)(COC)C1 CC1=C(F)CN(C(C2CC3(CC(NC(c4cnnc(C)c4C)=O)C3)C2)=O)CC1 Cc1ccsc1-c1ccc(-n2cc(-c3nnnn3-c3ccccc3)nn2)s1 C1(NC(C(C)OCCOC)=O)CN(C(=O)CCC2CC2(F)F)C2CCCC12 c1(C(=O)NC(C(C)(C)NC(C(CCC)C#N)=O)C)cccc2c1CCCC2 C12(NC(c3cc(C)c(OC)c(Cl)c3)=O)CN(C(=O)CC3CC3)CC1CS(=O)(=O)C2 CCC(CC(F)F)CS(=O)(=O)NCc1ccc([N+](=O)[O-])cc1F N1(C(CCCNC(CCOCCOCC)=O)=O)CCCC2CC12 N1(C(=O)N(C(C)(C)C)CCO)CCN(C(=O)C(CCF)c2ccccc2)CC1 CC1=C(C(=O)N2CCCOC(CCNC(=O)C(F)CC(C)C)C2)SCCO1 Cc1cc(N)ccc1C(=O)NCCNC(c1cc(O)nn1C)=O c1(N2CCC(C(C)(C)C)C(F)(F)C2)ccc(Br)c(S(=O)(=O)N2CCCC(F)C2)n1 C1(NC(=O)CCc2nc(O)n[nH]2)CCN(C(=O)CC2CCOCC2)CC1O C1(n2cc(CC(COC)O)nn2)CC2CCC(C1)N2C(=O)CCC(C)O N1(C(c2ccn(CC)n2)=O)C(C(=O)NCCN2CCNC(=O)C2)CC2CC12 c1(C(=O)NCC2(O)CC(NC(C=C3CCN(C)CC3)=O)C2)n[nH]c2c1CCCC2 n1(C(C)(C)C)cnc(C(=O)NCC2(CCNC(C3CC(C)(F)C3)=O)CC2)n1 c1(COC)cccnc1C(N1CCCC1CCNC(c1cc(C)no1)=O)=O CC(N(C)N1CCC(F)(F)C(F)(F)CC1)c1cccc(C2CC2)c1 Cc1nn(C)cc1C(=O)NC(C1CCN(S(=O)(=O)CC(C)C)CC1)C c1(C(=O)Nc2c(C(=O)OC)sc(C)c2)cccc2ccsc12 N1(C(CC2(C(=C)F)CCC2)=O)CCN(C(C2(C)COC2)=O)CC1C N1(C(c2cc(CN(C)C)on2)=O)CCC(C2OCCC2NC(=O)CC(F)F)CC1 O(NC(=O)CNC(=O)CSCCNC(=O)CC1CCC(C)C1)CC C(N=c1cccc(S(=O)(=O)NCC2CCOC2)[nH]1)C1(CCC)CC1 N1(C(C2(C)CCOCC2)=O)CCC2CN(C(c3cccc(F)c3)=O)CC2C1 CC12CCCC(C(=O)NCCC3(O)CCN(C(C4COC(=O)N4)=O)CC3)(CO1)C2 CC1(C)CN(C(=O)CCCn2ccnc2)CC1C(=O)NC1CCCSC1 c1(C2CC(c3n(CC)nnn3)(NCCC3OCCC3(C)C)C2)c(C)cccc1C C12(CNC(C3CC3c3ccco3)=O)CC(CN1C(c1ccc(C(F)F)s1)=O)C2 c1(C(N2CCN(C(C3C(C)C3C)=O)CC2CCO)=O)coc2ccccc12 Cc1cn2cc(NC(C3CCN(Cc4ccc(Cl)nn4)C3)=O)ccc2n1 c1(C(N2CC(CNC(c3coc(Cl)c3)=O)C2)=O)nccc2ncncc12 CCC(C)C(O)CC(=O)N(C(C)C(N1CCCCC1CO)=O)C1CC1 C(=O)(C1=NOC(C)(C)C1)N1CCCC(N(C(C2CS(=O)C2)=O)CC)CC1 N#Cc1ccc(C(O)C(=O)NC2CCC2NC(=O)C=CSCc2ccco2)cc1 CC(C)C(O)C(C)C(=O)NC(C)(C)CNC(=O)CCC1CCCO1 c1(CC(=O)NC(C)CCNC(c2cn(C)nn2)=O)ccc(Cl)c(F)c1 n1(CC)cc(C(=O)NC(C)CNC(C2CCC(CO)CC2)=O)c(C)n1 Cc1cc(Br)cc(Cl)c1C(N1CCOC(CNC(c2ncc(Br)cc2F)=O)C1)=O N1(C(c2c(C)c(F)cnc2)=O)CC(C)N(C(c2ncn(C(C)(C)C)n2)=O)C(C)C1 c1(C(C(=O)NCCOCC)N(c2cnn(C)c2)CC)nnc(C)s1 N1(C(C(F)=CCC)=O)CCC(CNC(=O)CSc2c(C)n[nH]c2C)C1(C)C C(CCO)(C(=O)NCC(C)(C1CCC1)NC(=O)CSc1ccc(O)cc1)N(C)C N1(C(C(C)Cn2ccnc2)=O)CCN(C(=O)C(=O)NCC2CC2)CC1CF c1(C(=O)NC(C(C)C)C(C)NC(=O)CSC(F)(F)F)cc2nc(Cl)ccc2o1 N1(C(Cc2c(OC)cccc2)=O)CCC(O)(C(C)NC(C2CC23CC3)=O)CC1 N1(C(CSCC)=O)CC(C(=O)Nc2cncc(C#N)c2)CC12CCC2 Cc1[nH]c2ccc(F)cc2c1C(N1CCN(C(=O)CC2CC23CC3)C(C)C1)=O N1(C(=O)CCOCC2CC2)CCC2(CCCCC2NC(C23CCC(C2)C3)=O)C1 c1(C(N2CCC(O)(C(=O)Nc3c(C)c(I)ccc3)C2)=O)c(Cl)cnc(Cl)c1Cl c1(C(N)=O)cc(C(=O)NCCC2CCCN2C(=O)CCNC(N)=O)cc(F)c1 C1(CNC(c2c(OC)nsc2)=O)CCCN(C(C2(C)CNC(=O)C2)=O)C1 N1(C(COCC)=O)CCCCC1CCN(C(=O)C(c1ccncc1)OC)C Cc1n[nH]c(C)c1CC(C)C(=O)NCC(O)CN(C)C(c1cc(F)c[nH]1)=O C#CC1CN(C(=O)CC=CC=C)CCN1C(c1cnc(C2CC2)o1)=O Cc1csc(C=CC(=O)NCC2CCC2NC(=O)CCCCc2cnn[nH]2)n1 Cc1cnc(C(C)NC(c2sccc2CNC(=O)COCC(C)C)=O)o1 C(=O)(C(C)S(C)(=O)=O)NC1C(C(=O)NC(C#C)CC2CCCC2)CCC=C1 c1(C(N(C2CCCCC2NC(C2CC2F)=O)C)=O)cc2n(c(=O)c1)CCS2 N1(C(C2CC(=C)C2)=O)CC(C2CCCCN(C(=O)CP(=O)(C(C)C)C(C)C)C2)C1 C1(N(CC(C)C)C(C2CCN(C(C(C)OCC#C)=O)CC2)=O)CC2CCC(C1)N2C C1(C(=O)NC2(CO)CN(C(c3c(C)n[nH]c3)=O)C2)C2CC2C2CC12 c1(CC(C)NC(CN(CC#C)C(C2CC2OC(C)(C)C)=O)=O)nncn1C C1(CCO)Cc2ccccc2CN1Cc1nscc1Br c1(CC)ccc(O)c(C(=O)NC(C)C(C)NC(c2cnnn2C)=O)c1 CC1CCCCC1OCCN(C(=O)OCCCNc1cccnc1O)C C1(C)(CC)CC(NC(=O)C2=CCCSC2)CN1C(c1ccc(=O)oc1)=O N1(C(C2(CNC(CCCCNC(C)=O)=O)CCCO2)=O)CCC2(CNC(=O)O2)C1 N1(C(CN(C)C)=O)CCN(C)C(C(=O)NCC2CCN(C3CC3)C2)C1 c1(C(=O)NCC(C)CNC(C2CCCN2C=O)=O)ccccc1S(C)=O C(c1ccc(C)cc1)=CC(=O)N(C1CCN(C(c2ccnc(OC)n2)=O)C1)CC C=C(C)CC(C(=O)NCCN1CCCOCC1)NC(c1c[nH]nc1Cl)=O CC1C(C)CN(C(C2(C)CN(C(=O)CCC3CCCO3)C2)=O)C1C Cc1nc2n(n1)CC(C(=O)NCCCCNC(C1CC3COCC3C1)=O)CC2 N1(C(=O)Nc2ccc(OCC)cc2)CC2CC(O)C1C2NC(c1cnsc1)=O C1(C(=O)Nc2ncc[nH]2)CC(F)CN1Cc1cccc(CO)n1 C1(C(C)NC(C(C)=C(C)C)=O)CN(C(c2cccc(Cl)c2)=O)CCO1 C1(CNC(CSCC(C)C)=O)CN2CCCCC2CN1C(c1cc(C#N)cs1)=O CCC(F)(F)CC(=O)N1CCC(N(C(=O)CCc2cnn(C)c2C)CC2CC2)C1 C(=O)(CC(O)CC(C)C)NCC1(COC)CN(C(c2c(C)ccc(Cl)c2O)=O)C1 N1(C(c2cn(C)[nH]c2=N)=O)CC(NC(C2(F)CC2)=O)CC12CCC2 c1(N2CCC(=C)CC2)nc(=NCC2CCCCC2C)[nH]c2ccsc12 Cc1nc2ccc(C(N3CCC(CF)(NC(C4CCC(C)(C)O4)=O)C3)=O)cc2o1 CCCC(C)(O)C(=O)N1CCC(NC(c2cnn3c2SCC3)=O)CC1 C(CC(C)(C)C(=O)NC1COCCN(C(=O)C=Cc2cccnc2)C1)SC C(C(=O)N(C)CC1CCCN1C(C1CCC(C(F)(F)F)CC1)=O)(C(C)C)SCC c1(C(=O)NCc2scc(CNC(Cc3c(C)noc3)=O)n2)nsc2ccccc12 N1(C(COC)=O)CC=C(C(=O)N(C2(c3cc[nH]n3)CC2)C)CC1 c1(C(=O)NC2(CNC(C=CCC)=O)CCC2)cc(C)cc(I)c1O C#CC1CN(C(c2cccc(F)c2CC)=O)CCN1C(=O)Cc1nocc1CC c1(SCC)ccccc1CC(N1CCSCC1CCNC(=O)Cc1ccsc1)=O C1(N(C(C(N2CCOCC2)C)=O)C)CCC(C(=O)NCC2CCC=CCC2)CC1 CC(CCN(C)C)C(=O)N1CCCCC1CC(=O)NCc1cc(C(N)=O)co1 N1(C(c2cc(CCC)[nH]n2)=O)CCC(C2CC(NC(c3sccc3Cl)=O)C2)CC1 CCS(=O)(=O)C(C)C(=O)N1CCC2(CC1)CC2C(=O)NCc1cccc(C)n1 Cc1ccc(CC(N2CCCC(NC(=O)C3=CSCCO3)CC2)=O)cc1C N12CCC(C(C)C1)C2=O.c1(C(C)C2CC2)cn(CCO)nn1 C1(NC(C(C2CC(NC(=O)C=C3CCCCC3)C2)F)=O)CCC(C2CC2)C1 c1(C(=O)NC(CNC(=O)Cn2cccn2)C2CC2)cc2cnccc2cc1F c1(CC(=O)N(C2CCC(NC(=O)CCC#N)C2)CC)coc2cc(OC)ccc12 c1(CC(=O)NC(C=CC(=O)N(CC#CC)CC#C)C)cnsc1 Cc1c(C(=O)NC(C)CC(=O)N(C)Cc2ccncn2)[nH]ccc1=O c1(CC)sc(=N)[nH]c1C(N1CC(OC)C(NC(C2(CCO)CC2)=O)C1)=O O=C(C1=Cc2ccccc2OC1)N1CCC2CCN(C(=O)C(F)CC3CC3)C2C1 C1(NC(CC2C(C)C2)=O)CN(C(=O)CCc2nncs2)Cc2ccnn2C1 Cc1ocnc1CCNC(C1CCC(n2cc(CCC3CCCOC3)nn2)C1)=O C(=O)(C1CCCc2nn(C)cc21)N1C(CNC(c2cccc(N(C)C)c2)=O)CC1 c1(C(=O)NCC2(OC)CCN(C(c3ccoc3C3CC3)=O)C2)ncc(N)cc1Cl CCCCCCCCC(F)C(=O)NCC(C)NC(=O)CCc1cnc(C)nc1O c1(C(=O)NCC2CC(O)CN2C(=O)CCC2CCC2)cccn2c(O)nnc12 c1(N2C(C)CC(NC(c3cnn(-c4ccncc4)c3)=O)C2)ncnc(Cl)c1F c1(C(=O)NCC2C(NC(C=CCOC)=O)CC2)c(Cl)cc(CO)cc1Cl c1(NC(C(C2CCN(C(c3ccc(Br)c(Cl)n3)=O)CC2)C)=O)cc(F)cnc1Br CCC(C)C(=O)C(=O)NC1CC(C)(NC(c2ccc(F)c(F)c2)=O)C1 c1(CCC(=O)N(C)CCNC(c2nccnc2C(N)=O)=O)c[nH]c2ccccc12 c1(OC)cc(C(=O)NC2(CO)CCN(C(=O)C(C)c3cncs3)C2)c(N)c(C)c1 C1(COCC(=O)NCC(C)NC(C2(c3nccs3)CC2)=O)CC(C)(C)CCO1 N(C(=NCCC(C)C)NCCNC(c1cc[nH]n1)=O)C1CC(C(C)(C)C)OCC1 N1(C(c2nc(CNC(=O)COC3CCC3)oc2)=O)CCC2(CC1)CC(O)C2 O=C(C1=NOC2(CCCN(C(c3c(F)cccc3Cl)=O)C2)C1)N1CCCC(F)C1 c1(OC)nn(C)c(Br)c1C(N1CCC(CNC(=O)C(C)(C2CC2)OC)C1)=O C12(NC(c3cnn(C)n3)=O)CCC(CN(C(c3ncsc3C(F)(F)F)=O)C1)C2 C1(N(C(c2cnn(CCOC)c2)=O)CC)CCN(C(c2cc(O)ncn2)=O)CC1 C(=O)(C(C(C)(C)C)n1cc(-c2nc(C)ncc2Cl)nn1)NC(C)=O.C12=CC=C(C=C1)C21CC1 n1(CC(N2CC(F)(CNC(=O)CSc3cn[nH]c3)C2)=O)nc(Cl)ccc1=O c1(OC)nscc1C(=O)NC1CCCC1CNC(=O)Cn1cnnc1O c1(C(N2C(C3(NC(C4C(=C)CC4)=O)CC3)CCC2)=O)ccc2ccsc2c1 C(=O)(CCCCCCCCC1CC1)NC1C(NC(C(N2C(=O)CCC2=O)C)=O)C1 N1(C(C2(CC)CCOCC2)=O)CCN(C(C2CC2(C)CC)=O)CC12CCC2 N(C(=NCCC(F)(F)C(F)F)NCC1N(C)CCCC1(C)C)CC(C)C N1(C(c2c(C)nco2)=O)C(CNC(C2C3CCC4C(C3)CC24)=O)CC2COCC12 c1(C(=O)NCC2CN(C(C=CSC)=O)C(C)C2)cc(Cl)c(F)cc1O c1(C(=O)NCC(CO)NC(C2C(C(=O)OC)C=C2)=O)nccnc1C(N)=O C1(NC(c2nc(NC(C)=O)sc2)=O)CCN(c2ncc(I)cn2)CC1O c1(C2(C(=O)NCC3C(CNC(CC(=O)NCC)=O)C3)CCC2)ccc(C#N)cc1 Cc1ccnc(-c2cn(C3(C(=O)NCC4CNC(=O)C4)CCOCC3)nn2)c1 n1(CC(=O)N(CCC(C(C)C)NC(=O)C(C)(C)CN(C)C)C)ccc(O)nc1=O Cc1scnc1C(=O)N(C1(C(=O)N(C)Cc2ncc[nH]2)CC1)C c1(C(=O)NCCC2(CNC(C3(CC(F)F)CCC3)=O)CC2)cnc(C(F)F)nc1 N1(C(CN(C)CC)=O)CCC2CCN(C(=O)Cn3ncccc3=O)CC12 c1(C(=O)NCC2(NC(c3ccc(OC)s3)=O)COC2)cc(OC)ccc1OC C1(CCC)(NC(C2CN3CCC2CC3)=O)CCCN(C(C2(CO)CC2(F)F)=O)C1 c1(N(C2CN(C(C(C)CCn3cccn3)=O)C2)C)cnn(C)c1C#N C=CC1CN(C(=O)CC(C)(C)N(C)C(C2CC2C)=O)CC1O c1(-c2cn(CCC)nc2)cccc(C(N2CCC(NC(C)=O)CC2)=O)n1 C1(C)(C(N(CC(CNC(CC2C(CC)C2(F)F)=O)(C)C)C)=O)CCCNC1=O N1(C(c2cncc(OCC)c2)=O)CCC(CNC(=O)CC=C(C)C)C1(C)C C12(CC)NC(=O)N(C1=O)C1CCC(C1)C(=O)NC2.C(C)(C)(C)OC(=O)NC1CC1 c1(CCNC(N(C(COCCOC)C)C)=O)ncc(C)o1 N1(C(C23CC(OC)C2C3)=O)CCC(CC(C)NC(c2cc(C(C)C)[nH]n2)=O)CC1 CCC(CC)C(F)C(=O)NC1CN(C(=O)C(C)CN(C)C)CC(F)(F)C1 O=C(CCCCCCc1cccs1)N1CCC(N(C(=O)C2=NOCC2)CCO)C1 c1(C(=O)NCCCCNC(c2cncc(Br)c2)CCO)ncncc1Cl C(=O)(CCCCCC#N)N1CCN(CCCNC(c2c(C)n(C)cn2)=O)CC1 c1(C(=O)NCC2CCCC(NC(C3(CC#C)CCC3)=O)C2)cc(C#N)ccc1N C1(CNC(c2cc(COC)[nH]n2)=O)CN(C(c2cnsn2)=O)C2(CCOCC2)C1 C12(C(N3CC(NC(C45CCC(C4)OC5)=O)C3)=O)CC3CC(C(=O)N1)C2C3 C1(CNC(c2cnn3c2OCC3)=O)CCC2(CN(C(C3CC(F)C3)=O)C2)O1 C1(CC(=O)N(CCCC)NC(CCC(=O)NCCC)=O)SC2=NCCN2C1=O c1(C(N2CC3OCC(NC(C4N(C)CCC4)=O)C3C2)=O)cc(Cl)cc2c1CCC2 N(C1CN(c2nc(O)ccc2C(C)C)CCc2ccccc21)C(C(C)OCC)=O C(=O)(CCCCCSC)NC1CCCN(CC(CC)C)C1 C=CCC(Cc1ccccc1)C(=O)OC1CCCN(CC(F)F)C1 CC(C)(O)C(F)C(=O)NC1(CCCNC(C2CC(n3ccnn3)C2)=O)CC1 C(=O)(C(O)CCC(C)C)NC(C(=O)NCC1(OCC)CC1)COCC C1(NC(C(c2ccccc2)NCCN(CC)CC)=O)COc2ccccc2C1=O C1(NC(c2nc(C)n(-c3ccccc3)n2)=O)CCC2CN(C(=O)C(C)C#N)CC12 N1(CC)CC(C(N2CCCCC2CC(=O)NCCCC(C)(C)OC)=O)CC1=O Cc1cnc(C(=O)Nc2cccc(O)c2Br)c[n+]1[O-] C(CCF)(C(=O)N(C)Cc1cn(C)nc1C)NC(CCc1cc(C)[nH]n1)=O c1(OC)cc(CN(C2CCN(C)C2C)CC2CN(C(C)=O)CCO2)ccc1C c1(CC(=O)N)cnc(Cl)c(Br)c1.Cc1nc(C(N2CCOCC2)C)sc1C(=O)NO c1(CCCC(=O)N(C)CCc2cccs2)nc2ccccc2[nH]1 c1(N(C)CC2C3CCCC23)ncccc1S(=O)(=O)NCC1(F)CCC1 N1(C(CCC)=O)CCC2(CC1)CN(C(=O)CCCC(C)CC)CC2CO N1(C(=O)CCc2ccc3c(c2)OCO3)CC2(CCCC2)OC2(CCC2)C1 N1(C(C2C(OCC)CC2)=O)CCCC(c2ccnn2C)CC1 C12(CNC(=O)CSC3CC3)CCC1CCN2C(c1csc(-c2ccc(O)cc2)n1)=O O=C(C#CC1CCC1)NCC1C2CN(C(=O)CC3(O)CCOCC3)CC12 c1(C(N2CC(F)(C(=O)NC(C(=O)OC)C3CC3)C2)=O)cccc2c1CCCC2 CC1CCN(C(=O)CNC(C2CC2NC(=O)CN2CCCC2)=O)CC1 C1(CC(=O)NCC(CNC(CCSCCCC)=O)CO)CCCC(C)(C)O1 c1(C(=O)NCC2C(NC(CC=CCC)=O)COC2)cc(C2CC2)cc(F)c1 N1(C(Cc2c(C)ccnc2)=O)CCC2(CC1)CC(NC(C1CNC(=O)N1)=O)CO2 C(=O)(C(O)CCCSC1CCOC1(C)C)NCc1cn(CC(=C)CC)nn1 C1(NC(C(CC)SC)=O)(CCCNC(C2CC2c2ccsc2)=O)CCOCC1 c1(CC)nc(C(=O)N(CC(CC)NC(=O)C(O)CC2CCCCC2)CC)cs1 C(=O)(CCCCCCC(=O)N1CCC(NC(C23CCC2C3)=O)C(C)(C)C1)OC n1(CC(N2C(CCN(C(C3C(=C)C3)=O)C)CCCC2)=O)cnc([N+](=O)[O-])c1 Cc1cc(=NC(=O)C(=O)N2CC(NC(=O)C(C)C(F)F)CC23CCCCC3)[nH]o1 c1(C(=O)NCCCCCCNC(C2(C)CC2(Cl)Cl)=O)ccnc2[nH]cnc12 C1(C2CCC2)(C(N2CCN(CCNC(CC3CCN(C)C3)=O)CC2)=O)CC1(F)F N1(C(C(C)CF)=O)CCC2(CCCCN(C(c3cc(Cl)ccn3)=O)C2)C1 c1(C(NOC(c2cnn(C)c2Cl)C)=O)ccc(CNC(C2CCC(C)CC2)=O)nc1 Cc1ccc(C=CCC(=O)N(C)CC2CCN(C(C3(C)CC4CC4C3)=O)C2)cc1 N(C1CCc2ccsc21)C(=O)Nc1n(C)nc(-c2ccsc2)c1 c1(C(=O)OCC)c[nH]c(=NCCCNC(=O)CN2CCN(C)CC2)s1 c1(C(=O)NC2C(CNC(C(n3ccc(C)n3)C)=O)CC2)csc2c(F)cccc12 c1(N(C)C)ncc(C(=O)NCC23CC2CN(C(=O)COCC2CCCC2)C3)cn1 c1(C(c2n(CC)nnn2)NCC2CC3(CCCCC3)C2)cc2n(n1)CCCCO2 C=CC(C)(O)C(=O)N1CCCC1C(N1CCN(C(C)=O)CC1)=O C1(C(=O)NC(c2ncnn2C(C)C)C)C=CCN(C(=O)C=C2CCC2)C1 CC(C)CCC(F)C(=O)NC(C)C(CO)NC(c1cnn2c1NCCC2)=O c1(C(N2CC3=C(CN(C(c4cncc(O)c4)=O)C3)C2)=O)cc([N+](=O)[O-])ccc1Cl N1(C(C(N2CC(CNC(C3(C)C(CC)CCC3)=O)C2)=O)=O)Cc2ccccc2C1 C(C(=O)NCC1(NC(C2CC2C2CCCC2)=O)CCC1)(C(C)(C)C)SC C1(NC(=O)CCC2CC2)CC(F)(F)CC1NC(=O)CN1CCC1 N1(C(C2CC(=C)C2)=O)CC(N(C)C(c2ccc(OCCOC)cn2)=O)C(C)(C)C1 c1(SCCN2CCN(C(C(N3C(C)CCC3C)=O)=O)CC2)cccc2ccccc12 C1(C2=CCCCCC2)(C(N2CCC(O)(C(C)(C)CNC(C3CCC3)=O)C2)=O)CC1 N1(C(c2c[nH]c(=N)o2)=O)CCC2(CCC2CNC(c2cncs2)=O)CC1 c1(C(N2CC3C(CNC(c4cccc(C)c4C)=O)(C3)C2)=O)c(C)nc2sccn12 C(CN=C(NC1CCOCC1)NC1CCC(C)(C)CC1)c1ncc(C)s1 c1(OCC)cnc(C(N2CC(NC(=O)CN3CC(C)(OC)C3)C(SC)C2)=O)cn1 N1(C(CC(CNC(c2ccc(C)o2)=O)C)=O)CCCC2(CCC2)C1 C(=O)(CC(C)C(F)F)NC(CC=CC)C(=O)NCCCCCCN(C)C C(C)(C)(CC(=O)NCC1CC(F)CN1C(c1cc(C(C)=O)oc1C)=O)OC C1(NC(CNC(c2[nH]cc(C(=O)OC)c2)=O)=O)CC2(CSC2)C1 N1(C(c2ccc(SCC)nc2)=O)CCN(C(C2(C)CCC(=O)C2)=O)CC1C1CC1 C1(CCC(=O)N(C)Cc2c(C)ncs2)CCCN(C(=O)C(O)c2ccco2)C1 CC(C)(C#N)CC(=O)NCc1c[nH]nc1C(=O)NC(C1CCC1)C1CC1 Cc1cc(F)ccc1C(O)C(=O)N1CCC1CNC(C1CCC(N(C)C)CC1)=O C12CC3(CCC3)C1OCCCN2C(C(N1CCCC(CCC)C1)C)=O.C(C)OC Cc1ncn(C)c(=O)c1C(=O)NCC(C1CCC1)NC(C1(C#N)CC2CC2C1)=O c1(C(N2CC(NC(CNC=O)=O)C(CC3CC3)C2)=O)nc2ccccc2[nH]1 N1(C(C2C(C)C2)=O)CCN(C)CC1CNC(=O)C(C)(C)c1cccs1 Cc1nsc(C)c1C(=O)NC1CCCC1CNC(C1CCCC1(F)F)=O Cc1cc(C(=O)N(CCCNC(C2C(C)C2(F)F)=O)C(C)C)c(O)c(Br)c1 c1(C(=O)NC(CC)CNC(=O)Cc2cscn2)cc(O)nc2ccc(F)cc12 c1(C(C)(C)C)c[nH]c2ncnc(N3CCC(F)C(COc4ccc(F)cc4)C3)c12 N1(C(CCCN(C)C(=O)NCc2cccc(O)c2)=O)CCC2(CC1)CC2N(C)C C12(NC(C3(C)CS(=O)(=O)C3)=O)CCCC1N(C(c1ccc[nH]1)=O)CC2 C1(CC(=O)NCC23CC(NC(=O)Cc4cnccn4)(C2)C3)CCC1C1CC1 C12(CC(N3CCCC(N(C(=O)CCc4nc(C(C)C)no4)C)C3)=O)COCC(C1)C2 O=[N+]([O-])c1cnn(CC2CC2)c1N1CCC2(C1)CC(F)C2 N1(C(c2c(C)cc(C)cc2N)=O)CCC2CCN(C(=O)C(C)S(N)(=O)=O)C2C1 CC#CCCCC(=O)NCC1CCN(C(=O)CC(C)(C)c2ccccc2)CC1C C1(NC(=O)CCN(C(=O)C=CC(F)F)C2CC2)CC2CC1CC21CC1 c1(CN(C(C(CC)=CC)=O)C)cnn2c1CN(C(=O)C(C)CC1CCCO1)CC2 N1(C(c2cccc(SC)c2)=O)CC2(CC(C(N3Cc4cncnc4C3)=O)CO2)C1 C1(C(=O)NCC(F)(F)Oc2ccccc2)COCC1c1ccccc1 N1(C(CCCCN(C(C(CC)COC)=O)C)=O)CCCC(C)(O)CC1 N1(C(c2ncc(C(=O)OCC)nc2)=O)CCN(C(c2cncs2)=O)CCC1C Cc1cc(N2CC(=O)NC3(CC3)C2)nc(=NCC(c2cccnc2)NC2CC2)[nH]1 CC1(C)OC2CC(C(N3CCC(O)(CNC(C4CCCCC4O)=O)C3)=O)CC2O1 c1(C(=O)NC2CN(C(c3c(OC)n(C)nc3)=O)CC2C)ccc2cnc(C)n2c1 C1(O)(CNC(C(N2CCOCC2)C)=O)CCN(C(c2cnc(O)o2)=O)C1.C1CC1 c1(C(=O)NC2CCC(C(=O)NC3C(OC)COC3)C2)ccn2nccc2c1 C1(CNC(C(CC=C)(F)F)=O)Cc2ccccc2CN1C(=O)CCc1ccoc1 C(=O)(C(C)(C(F)(F)F)N(C)C=O)NCC(C)Oc1cccc(Cl)c1.C(C)(C)(C)O C1(NC(C(C=C)(C)CC)=O)CCC2CC1CN2C(=O)CC12CC(C(=O)OC)(C1)C2 c1(OC)cc(C(=O)NCC2CC(NC(C3OCCC3C)=O)CCO2)cc(Cl)c1 Cc1ccc(C#N)cc1C(N1CCC(O)C(NC(=O)COCCCN(C)C)C1)=O Cc1cc(Cl)ccc1OCC(N1CC2(CC(NC(=O)CCCC#N)C2)C1)=O C1(C(=O)NCC2N(C(C3(C4(C)CC4)CC3)=O)CCOC2)CC12CCCCC2 C1(OCC)CC2CCCC(C1)N2Cc1cn(C)nc1C(=O)OC Cn1ccc(C=CC(=O)NCC2C(C(=O)NCC(C)(c3cccs3)N(C)C)C2)c1 c1(C(N(C(C)CN(C(=O)CCCF)C)C)=O)cc(Br)cc([N+](=O)[O-])c1 c1(CCC)ncoc1C(=O)NCC(C(C)C)NC(=O)Cn1cc(C(F)(F)F)nn1 c1(C(=O)NCCCC2(C)N=N2)cccc2ncccc12 N1(C(c2cc(CC)nn2C)=O)CCC2(C1)CN(C(=O)CC1(CO)CCC1)CCO2 Cc1cccc(O)c1C(=O)NCCCN(C)C(C1CCC(C2CC2)C1)=O CN(C)NC(=O)CCC(=O)NC12CC(CNC(c3cc(Cl)c[nH]3)=O)(C1)OC2(C)C C1(CNC(c2cn(C)nn2)=O)CCCCN(C(c2c(C(F)F)cccc2F)=O)C1 Cc1ccc(F)c(C(=O)NCC2(NC(c3n[nH]cc3F)=O)CCOC2)c1F O=C1c2ccccc2CN1OCc1ccc(-c2ccccc2)cc1Cl Cc1cnc(C(=O)NC2CC2NC(C2(F)CCCC2)=O)c(Br)c1 C(=O)(C1=CCCOC1)NCC(CNC(=O)C(c1ccc(F)cc1)C)OC C1(O)(C(N(C2CCN(C(=O)C(C)N3CC(C)C3)CC2)CC)=O)CN2CCC1CC2 C1(CC)CN(C(=O)CC(C)C2CC2)CCC1NC(=O)CCc1cccc(O)n1 C(=O)(CC(C)(C)C(F)F)N1CC(O)(C(C(N2CCC(OCC#C)CC2)=O)F)C1 C(C)(CC(C)CC(C)C)(c1n(C(CC)(C)C)nnn1)NCc1nnc(CO)s1 c1(OC)ccccc1C(CNC(c1ccn(C)c1C)=O)NC1(COC)CCCO1 c1(C(=O)OC)cc(C)n(CC(=O)NC2CCCC2NC(c2[nH]c(C)nc2C)=O)n1 N1(CCCC(=O)NCCCNC(c2n(CCC)ncc2)=O)C(=O)CCC1=O C1(C(=O)NC2C3CC(NC(Cc4cc(OC)ncc4)=O)CC32)COCCC1(F)F c1(N(CCCNC(C(C2CCCC2)OC)=O)C)ccccc1.C1(C)C(=O)N1 N1(C(CCOCCOC)=O)CC2(C(=O)Nc3cnc(F)c(C)c3)CCC1CC2 c1(C(C(=O)NC(C)(C)C)N(C2(C)CCC2)CC)cccnc1C c1(OC)cc(C(=O)N(CC(O)CNC(C2SCCS2)=O)C)c2occc2c1 C12(NC(C(CCC)c3cccc(Cl)c3)=O)CCCC1CN(C(c1cnsn1)=O)C2 c12ccc(Br)cc1C(=O)N2.c1(NC(C2C(C(=O)OC)C2)=O)cc(OC)ccn1 N1(C(C)C)CCC(CC(N2CCC(NC(=O)C(C)(C)c3ccsc3)C2C)=O)CC1 c1(NC(c2ccc(=NCc3ccc(CO)nc3)[nH]c2)=O)c(F)cc(Br)cc1F C1(CNC(C2(OC(C)=O)CC2)=O)CCCC(NC(=O)CC2(C)CCOCC2)C1 CON(CCC(=O)NCc1cc(O)cc(F)c1)C(=O)c1cc(C)nc(O)n1 N1(C(C2CCC(NC(C3CC(O)C3)=O)CC2)=O)CCn2ncnc2C1 N1(C(CC2(CC)CCC2)=O)CCCC(O)(CCNC(c2cn(C3CC3)nn2)=O)C1 C(C(=O)NC(C(=O)NC1CC1)C1(O)CCC1)(C(C)C)SC c1(C(=O)NC(CC)CNC(c2nncs2)=O)ccc(-c2ccncc2)s1 Cc1nc2cc(Cl)cc(C(N3CC(NC(=O)C4=CC(C)(C)C4)C(O)C3)=O)c2[nH]1 Cc1nc(CC(=O)NC2(CCNC(=O)CCc3cnn(C)c3)CC2)cs1 C1(O)(C(=O)NC2C=CC(C(=O)NCCC(=C)C)C2)CCSCC1 CC1(C)CC(NC(c2cnns2)=O)CCN(c2ncnc3c2SCCC3)C1 N1(C(C2C(C)OC(C)C2)=O)CCOCC(NC(=O)C(C)(C)CF)C1 CC1=C(C(=O)NC(C)(CNC(c2nnc(S)n2C)=O)Cn2cccn2)CCC1 C1(C(=O)NC2CC2NC(=O)CCSc2ccccc2F)(OCC)CCSCC1 CCC(CNC(C1CCC(O)CC1)=O)(CC)C(=O)N1CC(O)(c2nn[nH]n2)C1 C1(C(=O)OCCC2CC(NC(c3c(C)scc3)=O)C2)CCCCC1Cc1cc[nH]c1 N1(C(C(CNC(C2(CSC)CCC2)=O)O)=O)CCc2c[nH]nc2C1 N1(S(CC)(=O)=O)CCN(CCCN(S(=O)(=O)CC)CCO)CC1C C1(C(=O)NC(C)CNC(c2nocc2Cl)=O)CCC2(CC2)N1C(=O)OC(C)(C)C CC1CCN(C(C2CC2(C)C(F)F)=O)CC1N(C)C(c1cc(C2CCC2)[nH]n1)=O C(=O)(CC(C(F)F)n1cccn1)NCCCCNC(=O)C1=CCSC1 n1(CCC(=O)NC2C(C=C)CN(C(C3CCO3)=O)C2)c(C)nc2ccccc12 N(C(=NCCCc1cccs1)NC)CCC(=O)CC(C)C.C1(O)CCOC1(C)C C1(CCNC(CCOCCC)=O)CCN(C(C2NC(=O)OC2C)=O)CC1(F)F C1(C(N2CC(F)(CNC(c3c(C(C)C)onc3)=O)C2)=O)CCC2(CCOCC2)C1 N1(C(CCCCN(C(C)C)C)=O)CC(NC(c2cn(C3CC3)nn2)=O)CC(O)C1 c1(C(=O)NC2C(CO)CCN(C(C(COC)C)=O)C2)sc2ccc(Cl)cc2c1C N1(C(c2c(C)nc(CCC)s2)=O)CC2CC(C)N(C(=O)C=Cc3ncc[nH]3)C2C1 O=C1NCCN(C2CCc3ccc(F)cc32)C1CC1CC1 N1(C(C=CCCC)=O)CCC2CN(C(=O)C(C(C)CC)N(C)C)CC2CC1 c1(C(C)OC)ccc(C(=O)N(C2CN(C(c3ccco3)=O)CC2(C)C)C)c(O)n1 Cc1ccc([N+](=O)[O-])cc1S(=O)(=O)NC1(CC(=O)Nc2ccn(C)n2)CCC1 C1(OC)CCN(C(=NCc2cc(C)on2)NCC2(C)CCC(F)(F)CC2)C1 N1(CC(=O)NCCCNC(c2cncc(NC)n2)=O)CCC(C)(C)CC1 CC1(C(N2CC(O)(C(F)C(=O)NCc3cnccc3Cl)C2)=O)CCC(=O)C1 C12(C(=O)NCC3C4CN(C(C(c5ccccc5)C)=O)CC43)CC=CCN1CCC2 O=C(C1=CCCCO1)N1CCN(C(C2CCOCC2)=O)C(CO)C1 c1(CNC)cc(C(N2CC(C(=O)NCC3(N(C)C)CCC3)C(C)C2)=O)ccn1 Cc1ccnc(C(N2CC(C(N)=O)(CNC(=O)C(c3ccccc3)F)C2)=O)c1N C1(C(=O)NC2CCC(CCN)C2)(NCCN)Cc2ccccc2C1 C1(NC(Cc2c(CC)con2)=O)(CO)CCN(C(C23CCCC(CO2)C3)=O)CC1 C12(C(N(CC(=O)NCC(c3ccco3)O)CC3CC3)=O)CCC(C1)C2 C(=O)(C(O)CC(C)C)N1CCC(CN(C(C(CC)N(C)C)=O)C2CC2)CC1 c1(C(=O)NC2CC(CNC(=O)CCc3ccncn3)C2)cnn2c1OCCC2 C1(NC(=O)Cc2cncc(O)c2)CCN(C(=O)CC(O)C2CCCC2)C12CCC2 c1(C(N2CC(CC(=O)NCC3(C#N)CCC3)C2)=O)ccnc2c(Br)cccc12 N1(C(c2oc(C)c(S(C)(=O)=O)c2)=O)CCC2CC(C1)CN(C(C1CC1(C)C)=O)C2 N1(C(c2cc(C)[nH]c2C)=O)CCC(F)C(NC(=O)C(c2ccccc2Br)O)C1 C(=O)(CCCC(=O)OC)NC(C#C)CNC(=O)COC1CCN(C(=O)C2CC2)C1 CCC(CN(C(=O)C=CC(C)SC(F)F)C)NC(=O)CCC1CCCC1 N1(C(C(CCC)(C)C)=O)CC=C(CC(=O)N2CCCC(C(C)C)C2)CC1 c1(C(N2CCC(NC(C(C)(Cl)Cl)=O)C(CO)C2)=O)ccn2ncnc2c1 c1(C(=O)NCC2CCCN2C(C2CC23CCC3)=O)nc[nH]c2ncc(Br)c1-2 CCCC(CCC)C(=O)NCc1nocc1C(N1CCCCC1)=O C1(COC)CCN(C(C2(CO)CCN(C(c3ncccc3O)=O)C2)=O)CC1 CCC(COC)C(=O)NC1CCCC(NC(c2cc(C)n(C(C)(C)C)n2)=O)C1 N1(C(CC(COC)C)=O)CCCCCC1CNC(c1cc(C2(C)CC2)on1)=O N1(C(c2cc(C(=O)OC)no2)=O)CCCC(NC(=O)C(C)N(C)C)C1C c1(C2(C(=O)NC3C(NC(C=CC)=O)C3)CC2)ccc(OC(F)(F)F)cc1 C1(C(=O)NC(C(N2CC(NC(=O)NC)C2)=O)C2CCCC2)CCC(C2CC2)C1 O=C(CCCc1cnccn1)NCC1CC1NC(=O)C(F)=C1CCCC1 c1(NC(C=CC(C)NC(=O)CC2CC(O)C2(C)C)=O)cc(Cl)cnc1O O=C(NNC(=S)NCCCCCO)C(c1ccccc1)C1CC1 c1(C(=O)NCC(C)N(C)C(c2cccc(N)c2Br)=O)cc2ccc(F)cc2o1 Cc1cc(NC(C2CCCC(NC(=O)C#CC3CC3)C2)=O)n(-c2ccncn2)n1 c1(Nc2c(CNC(c3ccccc3)=O)c[nH]n2)ccc(C(=O)O)cc1O C(=O)(CN=c1cc[nH]cc1)N1CCN(C(C2C3CC4C(C3)C24CO)=O)CC1 CC1(CNC(c2ccccc2Cl)=O)CCCN1C(C12CCCC1C2)=O c1(NC(C2CC(O)CN2Cc2ccc3c(c2)OCO3)=O)cc(Cl)cc2[nH]ccc12 CCCS(=O)(=O)CC(=O)N(C1CCCC(NC(c2ccn(C)c2C)=O)C1)C C1(C(=O)NC2CCC(NC(c3c(CC)ccs3)=O)C2)Cc2cc(F)ccc2O1 C=C(F)C1(CC(N2CCC(C)(NC(=O)CCN3CCC3)C2)=O)CCC1 CC1C(NC(=O)C2=CCCCO2)CCCN1C(=O)CC(C)C1CCCO1 c1(N2CC(CC)N(Cc3[nH]c(C)cc3C)CC2)ncnc2cc(F)ccc12 C1(C(C)C)N(S(=O)(=O)CC(C)C#N)CC12CCCCC2 CCCCCN(CCC(=O)NC1CCC1NC(=O)C=CCOCCOC)C c1(-c2ccc(NCC(CC)(CC)c3ccccc3)o2)nc2ccccc2s1 c1(CC=CC=C)nnc(N2CCC(C(C)O)CC2)n1CC(=C)C.C1(C)CC1 C#CCCCCC(=O)NCC12CC(CNC(c3cccc(CC)n3)=O)(CO1)C2 c1(OC)cccc(COCC(=O)NCC2CC2NC(C2CC(C)N(C)C2)=O)c1 N1(C(CCCCC=CC)=O)CC(C)(CNC(=O)C(O)CN(C)C)CC1(C)C N1(C(=O)CC2(C(F)F)CCC2)CCN(Cc2cnc(-c3ccccc3)nc2)CC1 C(=O)(N=c1ccn(C2(COC)CC2)[nH]1)C1C(C=CNCC)CNC1 N1(C(CC(CC)O)=O)CCN(C(C2CC(Cl)(Cl)C2)=O)CC1CF c1(C(=O)OC(C=C)C(=O)OC(C)(C)C)cc2occc2[nH]1 C1(C(=O)OC)CCCC(C(=O)NC2C3CC2N(C(C2CCCC2(F)F)=O)C3)C1 C(C(=O)NCC(C)CNC(c1nc(C2CC2)cs1)=O)(C(C)C)SC c1(NC(CNC(c2n[nH]c3c2CCCC3)=O)CO)c[n+]([O-])ccc1[N+](=O)[O-] C1(C(C)C)CN(C(c2cccnn2)=O)CCN1C(=O)CCOC1CCC1 c1(C(=O)NC23CCCC2CN(C(C2CC=CCO2)=O)C3)cnc2sccn2c1=O N1(C(C2C(OC)(OC)CC2)=O)CCCC(N(C)C(c2cnn(CC3CC3)c2)=O)C1 N1(C(C(C(CC)C)O)=O)CCC(C(=O)NCC(F)(F)F)=C(F)C1 N1(C(C(C)CN(C)C)=O)CC2(CNC(=O)Cn3cnc(C(F)(F)F)c3)CC1CO2 C(=O)(CCCCCCn1cnnn1)N1C(CN(C(C2CCCOC2)=O)CC)CCC1 c1(C(=O)NCC(C)(C2CC2)NC(c2c(C)ccnc2)=O)c[nH]c(=N)cc1C N1(C(c2cccc(C(C)=O)c2C)=O)CCCN(C(=O)C(C)N2CC(C)C2)CCC1 CCC(CCC(=O)NCCC(=O)N(C)C)NC(C1CC(=O)C1(C)C)=O c1(OCC)ccc(C(=O)NC(C)(CNC(=O)CC2CC=CCC2)C(C)C)cc1Cl N1(C(CC(C)F)=O)CCCC1(C)C(=O)NCC1C(C)C1C C1(C(=O)NCC2(CNC(c3ccc(SC)o3)=O)CCCC2)CCCCC1O c1(C(=O)NCC(CC)NC(=O)C(c2ccc(C)cc2)C)nn(C)cc1C C1(CC)CN(C(c2cscc2OC)=O)CCC1NC(=O)C=CCF CCCC(C)C(=O)N1CC(NC(=O)CNC(=O)CC(C)(C)C)C1 [N-]=[N+]=NCCCC(=O)NCC1CCCCC1NC(c1c[nH]nc1C1CC1)=O Cc1cccn(CC(N2CCN(C(c3cnn(C4COC4)c3)=O)C(C)C2)=O)c1=O N1(C(C(C(C)C)F)=O)CCC(O)C(NC(=O)C(C)(C)C2CC2)C1 S(=O)(=O)(c1cccnc1)N1CC(C(N2CC(C)N(CCO)CC2)=O)C(O)CC1 c1(COC(c2ccc(NCc3nc(C)sc3)cc2)=O)cc(O)cc(Cl)c1 c1(CC)ccc(C(=O)C(=O)NCC2CC(NC(C3CC3c3ccn(C)c3)=O)C2)s1 N1(C(C(C)(CN)C2CC2)=O)CCN(C2CCCCC2)C(=O)C1 c1(N(CCCNC(=O)C=CC(=O)NC2CC2)C)ncnc2cccc([N+](=O)[O-])c12 C(=O)(C1Cc2ccccc21)NCC1C(NC(C2(C#C)CCCC2)=O)C1 N1(C(C(=O)NCCOCCCC)=O)CC2COCC(C1)C2NC(=O)C1=CCSC1 C12(C(N3CC(COC)(NC(c4cnc(Cl)s4)=O)C3)=O)CCC(C1)OC2 C1(C(N2CC(CNC(C3CCCNS3(=O)=O)=O)C2)=O)CC2CCC(C1)C2O C1(N(CC#C)C(C2CCCO2)=O)CCN(C(=O)COCC(C)(C)C)C1 c1(CNC(NCCC=CC=C)=NC)ccc(Br)cc1Cl C1(NC(c2cc(C)nc(O)c2)=O)CC2CCC1N(C(C1(F)CC=CCC1)=O)C2 N1(C(c2ccc(SC)cc2)=O)CC2CC(C)N(C(c3cccc(CO)n3)=O)C2C1 C1(CC)CN(C)C(=O)CN1C(C1(NC(=O)C(F)=CC2CC2)CCC(C)(C)C1)=O C(C1c2ccccc2CN1C(=O)OC(C)(C)C)NC(c1c(C(C)O)cccc1)=O N1(C(C(C)(C)C)=O)CCCC2C1CCN2Cc1ccc(F)nc1 N1(CC)CC(C(=O)NCCOCCNC(c2cnnc(C(F)(F)F)c2)=O)CC1=O CC1=NN(C)C(=O)C1CC(=O)NCCOCCN(C)C(c1nccc(Cl)c1F)=O N1(C(CCCCN(C(=O)C(O)CC2CCCC2)C)=O)C(CO)CCC12CCC2 c1(OCCC2CN(C(c3c(C)onc3)=O)C2)ccc(NC(C2CC2Cl)=O)cn1 C1(CNC(C(c2cnn(C)c2)OC)=O)CN(C(=O)CCC2CCC2)CC1(F)CO c1(C(N(CC(CN(C(C2(CCOC)CC2)=O)C)O)C)=O)ccc(CO)o1 C(=O)(CC(C(F)(F)F)P(C)(C)=O)NCCN(C(C(CC)C#N)=O)C1CC1 C(C)(C)(CC(=O)NCC1CN(C(=O)C(F)(F)c2cncs2)CC1C)OC N1(C(CC(C)(C)OC)=O)CC(CO)C2(C1)CN(C(=O)CC1CCCCC1O)C2 c1(NC(=O)NC(C)(C)C(O)c2ccccc2)c[nH]c2ccccc12 C1(N(CC#C)C(c2[nH]ccc2C)=O)CCN(C(C2SCCC2C)=O)CC1 Cc1nsc(N)c1C(=O)NCC1(CC(=O)NCC2CC(=O)N(C)C2)CC1 n1(CC(=O)NC(C)CCCNC(=O)CCc2ccc(F)cc2)ccc([N+](=O)[O-])n1 Cc1cc(C(N2CCC(OC3CCCC3)C2)=O)nc(C)c1.c12ccncc1OC2 N1(C(c2cnc(CCC)s2)=O)CCCCC1C1CCN(CC=CCOC)C1 CCC(CC)(CO)C(=O)N1C(C(=O)NCCNC(=O)C(C)C)CC1C c1(C(N2CC(COC)(NC(=O)C(N)=O)C2)=O)ccc(C)nc1Oc1ccccc1 N1(C(COCC)=O)CC(NC(c2cccc(Cn3cccn3)c2)=O)C(C2CC2)C1 Cc1ccc(C(CCO)NC(=O)CCC2CN(C(=O)CN(C)C)CCO2)cc1 CCC(C)C(C(=O)NCCn1ncccc1=O)N(C(=O)Cn1cnnn1)C C(=O)(C1c2ccccc2CN1C(c1ccccc1Br)=O)N(C1CC1)CC Cc1cccc(Br)c1C(=O)NC1CCCC(C(=O)NCc2ccc(F)cc2F)C1 Cc1ccc2c(=NC(=O)C3CCC4(CCN(C(=O)CNC=O)CC4)C3)[nH][nH]c2n1 C(=O)(C(C)(O)CC(F)F)N(CCNC(c1c(C)cn(C)c1)=O)C C(=O)(CCN(OC)C(=O)CC1(C)CCN1C(=O)CNC(C1CC1C)=O)OC Cn1nc2ccccc2c1NC(=O)NCCn1nccn1 C1(CNC(C2CC3C=CC2C3)=O)CC2CC1CN2C(=O)Cc1cnoc1 c1(OC)cccc2c1CN(C(C1CCN1)=O)CC(C)(C)O2 CC1=C(C(=O)NCC2(O)CN(C(=O)C3Cc4ccc(Cl)cc43)C2)CCC(C)(C)C1 CC1=C(C(=O)NC2(CO)CN(C(c3nnn(C(C)(C)C)n3)=O)C2)S(=O)(=O)CCO1 CCCC(CCC)=CC(=O)NC(CCNC(C1(N(C)C)CCCCC1)=O)C(C)C N1(C2C(CNC(c3cncc(-n4ccc(C)n4)n3)=O)CCC2)CCCN(C)CC1 Cc1ccn(C)c1C(=O)NCCC1(O)CCN(C(=O)CNc2nccs2)C1 N1(C(C2N(C(c3c(C)con3)=O)CC(F)(F)C2)=O)CCCC2(C=CCO2)C1 C12(CC)CCC(C(N3CCC(NC(=O)Cc4cccc(F)c4)CC3)=O)(CC1)CO2 CC(C)CC(=O)C(=O)NCc1ccc(C(=O)NCC(C)(O)C(F)F)o1 c1(C(N)=O)cc(C(=O)NCCCNC(=O)C=C2CCCCC2)n[nH]1 CCCCC(C(=O)N(CCC(C)C)C)NC(C1CCCN1C(C)=O)=O N#Cc1ccc(S(=O)(=O)N2CC3CC3(CO)C2)cc1NCC1CCCS1 CCC(C)C(C(N)=O)NC(C1CCN(C(=O)Cc2ccn(CC)n2)CCO1)=O c1(C(=O)NCC(CC)N(C)C(c2cnc3[nH]nnc3c2)=O)n[nH]c2c1CCCC2 C(CCCC(CO)NC(c1ncc(Br)cc1C)=O)NC(C(C=C=C)C)=O N1(C(C23OC(C)C(C2)C3)=O)CCN(C(=O)Cn2cc(C#N)cn2)C(CO)C1 N1(C(c2[nH]c(=NC)sc2)=O)CCN(C(c2cccc(F)c2)=O)C(CC2CC2)C1 CCCC(CCCNC(=O)C(C)CCCOC)NC(=O)Cc1c(C)nn(C)c1C C1(C(=O)NC(CC)CN(C(=O)CCCCCOC)C)CCC2(CCC2)CO1 C1(NC(C(CC)(C)CCC)=O)CCC(F)(F)CC1(C)C N1(C(C2(CC)CCCC2)=O)C2CCC1CN(C(C1CC1C1CC1)=O)C2 C(=O)(C1=C(Cl)CCC1)NCC1(F)CCN(C(CCOC)=O)C1 C1(CCC(=O)C(F)(F)CC2CCNCC2)CCc2ccccc2C1.N N1(C(C(C)NC(C)=O)=O)CC2C3CCC(C2C1)N(C(=O)CC1CCC(=O)O1)C3 CC(C)C(O)C(=O)N1CCC(NC(c2cccc(C(=O)OC(C)C)n2)=O)C1 C12(NC(CC3CC(OC)C3)=O)CCCC(CN(C(c3cccc(Cl)c3F)=O)C1)C2 C1(C)(NC(CCC2CCN(C(c3c(C)nsc3)=O)C2)=O)CCCC1(F)F C(=O)(CC1=NNC(=O)C1)N1CCC(N(C(=O)COCCCC(C)C)CC#C)C1 N1(C(c2c(CNC(=O)CC3OCCCO3)occ2)=O)CCOC2CC12 C1(C(=O)NCC2CN(C(Cc3cccc(OC)c3)=O)CC2O)OCCN(C)C1=O C(CNC(=O)CCn1ncn(C)c1=O)(C(C)C(C)C)NC(C)=O N1(C(C)=O)CS(=O)(=O)CC1C(=O)NCC1CCCN(C(c2ccc(C)cn2)=O)C1 N1(C(C2(C)CC2c2ccccc2)=O)CCN(C(=O)C=CBr)CC2(CC2)C1 C(CN(C)C)(CN=c1ccc(C(=O)OC(C)(C)C)c[nH]1)OCC C=CCC(CC=C)C(=O)N1CC(CNC(=O)COCC)OC(C)(C)C1 c1(N2CCC(CNC(C(C(CC)(C)C)O)=O)C2)nc2c(cc1C#N)CN(C)CC2 C(CCC)(C(=O)NCc1ncoc1C1CN(C(c2cnc(C3CC3)o2)=O)C1)=CCC N1(C(C(=O)N(C)C)=O)CCCC(F)(CNC(=O)Cc2ccnn2C2CCCC2)C1 Cc1cn(CC(N2CC3CC(NC(C4C(C)C4C)=O)CC2C3)=O)c2ccccc12 CC(C)C(C)CC(=O)NCCS(C)(=O)=O.C123CC1CN(C2)C(=O)CCCC31CC1 Brc1cnc(N2CCN(CCc3cccc(-c4ccccc4Br)c3)CC2)c(Br)c1 N1(CC(=O)NC(C)CCNC(=O)CCOC2CCC2)CCCC1=O C12CCN(C1C)C(=O)CN2CC1CC1.C12CCCN1C2=O.C#CCOC Cc1cnc(Cl)cc1NC(C1C2CC1N(C(c1ncoc1C)=O)C2)=O C(=O)(CCCC(CC)NC(=O)CSCCOC)NCCC=C=C C1(C(=O)NC(C2CCCC2)C#C)CCN(C(c2c[nH]c(C)c2)=O)C1 c1(C(=O)NC(C)CNC(=O)C(C)OC2COC2)cn2ccc(CO)cc2n1 CN1CCCC1CCC(=O)N(CC(N1CC(C)(N(C)C)C1)=O)C1CC1 CCC(CN=c1[nH]ccn2ncc(I)c12)OC N1(C(c2c(CC)n(CC)nc2)=O)CCC2C1CCCN2C(C1CC(N(C)C)C1)=O N1(C(c2cc(C)c(C)[nH]2)=O)CCC2(CCC(NC(C3(F)CCC3)=O)C2)C1 CC1(C)CCCC(O)(C(=O)NCC2(O)CCCN(c3cc(C(N)=O)ncn3)C2)C1 C12(CC(=O)NCCCC(C)NC(C3(C(CC)=O)CC3)=O)COC(C)(C1)C2 N1(C(C(C)N(C)C)=O)CCCC(CCNC(=O)C=Cc2ccc(Br)o2)CC1 CC(C)(C)CCC(F)C(=O)N1CC2CN(C(c3ccn(C4CC4)n3)=O)CC(C1)O2 C1(C)(CC)CC(CO)(NC(C2(C)CC=CCC2)c2nnnn2C2(C)CC2)C1 c1(C(=O)NC(C2CCN(C(C(CC#C)O)=O)CC2)(C)C)cn(C)c(=O)n1C C=C1CCN(C(c2ccc(C)nc2O)=O)C(C(=O)NCC(C)(F)C(C)C)C1 Cc1ccc(F)c(C(=O)NCC2CC3CC3N2C(=O)Cc2nc([N+](=O)[O-])n[nH]2)n1 n1(C2(C(=O)NC(CNC(C3(COC)CC3)=O)C)CC2)cc(Cl)cn1 C(=O)(C1=C(C)CCOC1)N1C(C)CC(NC(c2c(OC)ncc(F)c2)=O)C1 C1(F)(CNC(C(CSCC)NC(=O)C(CC)N(C)C)=O)CCOCC1 N1(C(c2nncn2CCOC)CC)CCCC(C(N2CC(C)OC(C)C2)=O)CC1 C1(CSC)CCC(NC(c2cccc(Cl)n2)c2nnnn2C(C)C)CC1 C(=O)(CCC(=O)C1CC1)N1CCC(C(C(=O)NC2(COCC)CC2)C)C1 c1(CC(=O)NC(C(C)NC(c2ccn(C)n2)=O)CO)ccc(O)c(Cl)c1 N1(C(C(CC)(C)F)=O)CC2(CCN(C(=O)CNC(C3CCOCC3)=O)C2)C1 C(=O)(CCCC(F)(F)F)NC1C(NC(C(C)(C)c2cc[nH]n2)=O)C1 CCC(C)(CO)C(=O)N1CCN(C(=O)C(C(C)C)NS(C)(=O)=O)CC1 c1(ONC(CN(C(C(C)C)C(=O)NO)C)=O)cc2ncccn2n1 C1(C(N2CCC(Cl)C2)=O)C2CC(F)C(C2)N1C(c1c(F)ccc(O)c1F)=O C(CC(=O)OC)(C(F)(F)F)C1CC(CC(N2CCC(COC)C(C)C2)=O)C1(C)C C1(C(=O)NC2CC(NC(CC3(COC)CCCC3)=O)C2)C2CS(=O)(=O)CC12 C(=O)(C(O)CCNC=O)NCC(C)(C)Cn1cc(C(C)(C)CO)nn1 C(=O)(CCCN(C)N=O)NCC1(CNC(C(CC)(C)F)=O)CCCC1 c1(C(N2CCC(NC(C(CC=C)(C)C)=O)C2C)=O)ncc2[nH]ncc2n1 c1(C(C(=O)NC)N(CC)Cc2ccoc2)cc(C)sc1C N12CCC(CC1)CNC(=O)C1C(C1)C2=O.C1(C(=O)OC)CCC1CN(C)C n1(CC=C)nnnc1C(C(C)C1CCCC1)Nc1cnn(CC2CCCC2)c1 S(=O)(=O)(c1ccc(C(N2CCN(C(C3CC34CC4)=O)C3CCC23)=O)o1)NC [N-]=[N+]=NCCCC(=O)NCCC1CC(C(=O)NCCc2cccs2)C1 c1(C(N(C(C)CNC(=O)Cn2nnnc2C)CC)=O)cc(Cl)ns1 O=C(C1CCc2ccc(Cl)nc21)NCC1CC2(CCN(C(C3CC3F)=O)CC2)C1 C1(C(=O)NC(CCOC)C(=O)NCC2CC=CCN2C(C)=O)CN2CCC1CC2 C(=O)(CC(O)CC(C)(C)C)N1CC(C(=O)NCCCCCCC=C)N(C)CC1 c1(C(=O)NC(C2CCN(C(=O)CCC(=O)N(C)C(C)C)C2)C)nc(=O)n(C)[nH]1 N1(C(C=COCC)=O)CCC(NC(c2nc(C3CC3)ncc2Cl)=O)C(C)C1 Cc1cc(C)c(C(=O)NCCC2COCCN2C(c2cc(C)sn2)=O)cn1 C1(NC(=O)C(F)F)CCCCCN(C(C2CC3OC2C2CC32)=O)C1 O=S(=O)(c1ccc(NC2CC3(CCC(F)(F)CC3)C2)c(Br)c1)NC1C=CCCC1 c1(C(=O)NCCC(C)N(C(C(CC2CC2)OC)=O)C)nn(C)cc1SC C(C(C)N=c1cc(NCc2cnccc2C)nc(C(F)(F)F)[nH]1)OCC CC(C)(CO)C(=O)N1CCC(F)(CNC(c2csc(-c3cn[nH]c3)n2)=O)C1 C(=O)(C(C)(C)C(=O)N1CCC(C(F)F)(CNC(C2(S(C)(=O)=O)CCC2)=O)C1)NC c1(C(N(CC(C)NC(c2[nH]cc(CC)c2)=O)C)=O)cccc2ccc(C)nc12 Cc1nc(C(=O)NCC(C)N(C(=O)C#CC(C)C)C)nn1-c1nc[nH]n1 n1(C(C)C)cncc1CC(N1CC(C)(c2cn(C3CCC3)nn2)C1)=O C(=O)(C(C)CC#N)N1CC(CC(C(=O)NCc2cnc(C)s2)F)C1 c1(C(=O)NCC2C(NC(=O)C=CC3CCC3)COC2)ccc(C(F)F)nc1 C1(NC(CCC(C)OC)=O)CCCCN(C(=O)C=Cc2cccc(O)c2)C1 Cc1cc(=NC(C)c2csc(C(F)(F)F)n2)[nH]c(=NCCc2ocnc2CO)[nH]1 C(=O)(C(N)(C(F)(F)F)c1ccc(OC(F)(F)F)cc1)NCC(c1cn(C)nc1)=O C(=O)(C(F)(F)C(O)C(C)C)NCCOCCNC(c1ccc(C)nc1C(C)C)=O C1(C(N2CCCC(CN(C(c3c(Cl)cc(C)s3)=O)C)C2)=O)CC2(C1)CC(F)C2 N1(C(CNS(C)(=O)=O)=O)CCC2(CNC(C3CC(=O)N(O)C3)=O)CCCCC12 c1(C(N2CC(NC(CN(C(C)=O)C)=O)C2)=O)ccc(C(F)(F)F)c(Cl)c1 C(=O)(C(F)C1=CCCCC1)N(C)CCC1CCN(C(c2csc(CO)n2)=O)CC1 C(=O)(CC(C(F)(F)F)NC(=O)CCN1CCC1)Nc1cn(CC(C)C)nc1 Cc1c(NCCC2CCCO2)ncnc1N1CCC(c2cc(O)n[nH]2)C1 C1(C(=O)NCCC(C)CCNC(C2(C#N)CC2)=O)CCCC(F)(F)CC1 CC(C)(CC(F)(F)F)C(=O)NCCC1CCCCN1C(=O)CC(F)F C#CC1CCC(C(N2CCC(NC(=O)C(C)=C3CCC3)C(F)C2)=O)CC1 c1(OC)ccc(C(C)(C)C)cc1CNCc1nc2c(o1)CCSC2 C1(NC(C23CCC(C)(CC2)OC3)=O)CC(C2CCN(C(C3CCOC3=O)=O)C2)C1 c1(C(N2C(c3cn(NC(c4ccc(OC)o4)=O)nn3)CCC2)=O)nccc(Cl)c1Cl N1(C(c2onc(CC)n2)=O)CCCC(C2CN(C(=O)CN3C(C)CCC3C)C2)C1 Cc1oc(C(C)(C)C)cc1C(=O)NC1(CCNC(=O)CC2CC23CC3)CCCC1 c1(C(N2CCC(CCC(=O)NC(C3CC=CCC3)(C)C)C2)=O)ccc(O)nn1 c1(C(=O)NCC2N(C(C(C=C)O)=O)CC(OC)C2)cc(Cl)cc(Cl)c1Cl N1(C(C(CCC)(C)C)=O)CCN(C(=O)CC2(C)CCCCC2)CC12CCC2 CN1C(=O)CCC1C(N1CCC(NC(c2ccc(CO)nc2)=O)C1C(F)F)=O Cc1cc(Cl)c(C(=O)NCC2CC2NC(=O)C(O)CC(F)F)cc1Cl CCCC(C)(O)CC(=O)NCC1(C)CCCN(C(c2sccc2CC)=O)C1 c12cccnc1CNC2=O.C1(COCC#C)CCCN1C(C1CC=CC1)=O Cc1cc(F)sc1C(N1CC(F)CC1CNC(=O)CCC1CCCC1)=O c1(CNC(CC2OCCN(C(C(C(=O)OC)(C)C)=O)C2)=O)cc2ccccc2o1 c1(OC)cccc2sc(C(N3CCC3CNC(C3CCC4(CC3)CC4)=O)=O)cc12 C1(OC)CC(CNC(=O)CC(C)(C)C)N(C(C23CCC(C2)C3)=O)C1 C1(N(C(C(CN(C)C)O)=O)C)CN(C(=O)Cc2ccnc(O)c2)CC12CC2 CC(C)CCCC(=O)N1CCC(n2cc(C(=O)Nc3ccccc3N)nn2)CC1 c1(C(=O)NCCC2CCN(C(C(F)=CCC)=O)C2)ccc([N+](=O)[O-])cc1CC C12CC3(C1)CN(C3)C(=O)C2.C1(OC(C(C)C)=O)CCN(C(=O)N)C1.c1(C)cnc[nH]1 c1(C(N2CCC(CN(C)C(c3coc(Cl)n3)=O)C2)=O)cc2c(Cl)cccn2n1 N1(C(C(CC)=CC)=O)CCC2C(C1)CN2C(c1ccn(C2CC2(F)F)n1)=O C(c1ncccc1C)=CC(=O)NCCOC1CCN(C(CN(C)CC)=O)CC1 C1(c2cn(CC3OCCN(C(=O)CSC4CC5CCC4O5)C3)nn2)CCCC(F)(F)C1 CC(CCS(C)(=O)=O)(c1nnnn1C1CC1)NCCC(C1CCOCC1)O c1(C2(C(=O)NC(C)CCCNC(=O)Cn3nnc(=O)[nH]3)CC2)cccc(F)c1 C12(NC(=O)CCOC3CC3)CC1CN(C(c1ccccc1-n1cncn1)=O)C2 N1(C(c2cc(SC)oc2)=O)CCCC(CNC(C2(C)CCC3CC3C2)=O)CC1 CS(=O)(=O)c1cc(C(N2CC(NC(C3CC3c3ccccc3)=O)C2)=O)ccc1F Cc1cc(C(=O)NC2CN(C(C3(C)CCCN3C)=O)C2)c2nccc(C)c2c1 Cc1nc2c(C(N3CCN(C(=O)CC(C)(C)C)C(C(C)(C)C)C3)=O)ccnc2[nH]1 c1(C(=O)NC2CC(C)(Nc3cc(Cl)nc(C(F)(F)F)n3)C2)cc(Cl)nnc1Cl C1(C(=O)O)CC2(CCCC2)CCN1C(=O)CCC(=O)c1cccc(N)c1 CC1CCC(CNC(C2(C)CC2)=O)N(C(=O)C=CI)C1 C(=O)(C(F)(F)C(C)O)N(CCCNC(c1occ(C)c1C)=O)CC1CCCC1 C1(NC(c2cc(C)oc2C)=O)CN(C(c2c(C)cccc2Cl)=O)CC1C1CC1 N1(C(C(C)N2CCC2)=O)CCN(C(C)CNC(C2(C)CC(C)(C)C2)=O)CC1 Cc1cc(C(N2CC(C)(OCC(N3CC(C)CC3C(N)=O)=O)C2)=O)cnc1C C1(COC)(NC(c2nncs2)=O)CCN(C(C2CC2C#N)=O)CC1 c1(-c2cn(C(C(N3C(C(=O)OCC)CCCC3)=O)C)nn2)cc(C)cnc1F N1(C(C(=O)Nc2ccc(C)cc2)C)CCN(C(=O)CCF)C(C)C1 N1(C(C(C(C)(C)C)NC(C)=O)=O)CCN(C(=O)C#CC2(C)COC2)CC(O)C1 C1(NC(C(C=C)(C)CCOC)=O)CC1C1CCN(C(=O)C=CCN(C)CC)CC1 C(CCCCCC(=O)N1CC(O)CC(C)(C)C1)NC(C(CC)=CC)=O C(=O)(CS(=O)C(F)(F)F)NCC1(O)CN(C(C(CC=CC)CC)=O)C1 C(=O)(C#CC1(C)CCCO1)NC(CNC(CCNC(=O)OCC)=O)(C)C1CC1 Cc1oc(C(C)(C)C)cc1C(N1CCC(CF)(NC(=O)C(C)CF)C1)=O N1(C(CC2N(C)CCCC2)=O)Cc2ccccc2C2(CC2)C1 N1(C(C(CN(CC)CC)F)=O)CCCCC1CN(C(=O)CC(=O)N(C)C)C CC(=O)C(C)CC(C)C(=O)N1CCCC(C)(NC(C2CCC(C)CC2)=O)C1 N1(C(C(C)n2ccnn2)=O)CC2(C(N3CCSC4(CCC4)C3)=O)CC1CCO2 N1(C(CCc2c(C)nccc2)=O)CCN(C(C2CCCCC2)=O)C(CC(F)F)C1 Cc1ccoc1C(=O)NC1(C)CN(C(C2(C)CC2(F)Cl)=O)C1 C12(C(=O)NCCCC=CC)CCN(C(=O)COC)CCC1C2 CCCS(=O)(=O)C(C)C(=O)N1CCN(C(=O)CCSC2CCCC2)CC1CCO C1(O)(C(N(CC(O)CNC(C2CCOC2c2nccn2C)=O)C)=O)CCCCC1 C(=O)(C1=CCc2ccccc21)N(CCNC(C=Cc1c(C)ncs1)=O)C N1(C(CCCC)=O)CCC(CNC(=O)C(=C2CCCCC2)F)C(O)C1 C1(CNC(C2CC3(CSC3)C2)=O)CC2(CCN(C(=O)COC3COC3)CC2)CO1 c1(C(C)NS(C2CCC(OC)CC2)(=O)=O)ccc(C2=CCNCC2)cc1 Cc1ccc(F)c(CCN(CCC#N)C(C2C3C4CCC(C4)C23)=O)c1 C1(C)(OC)CC(NC(C2CCCN(C(=O)C=Cc3ccncn3)CC2)=O)C1(C)C N1(C(C(CC)NC(C)=O)=O)CCCN(CCNc2ccccn2)CC1 C1(CNC(=O)Cc2cscn2)CCC2(CCC2)C1NC(C1CCS(=O)CC1)=O C(O)(CCNC(=O)CCC(N1CCCC(CC(C)C)C1=O)=O)(C(F)(F)F)SC N1(C(c2cncc(C)n2)=O)CCN(C(c2ccc(F)c(F)c2F)=O)CC12CCC2 C1(C(N(C(C)C)CCNC(C2COCOC2)=O)=O)CCOCC1(C)C CCC(C)(O)CNC(=O)C(CN(C)C)NC(c1cn[nH]c1)=O N1(C(C2(C(=O)OCC)CCO2)=O)CCOC(CCNC(=O)C=CC=C(Cl)Cl)C1 N1(C(c2c(C)cncc2)=O)CCCC(C2CCN(C(C3OCCO3)=O)CC2)C1 CC(C)C(C)CNC(=O)C(O)CNC(C1(n2cnnn2)CC1)=O C1(NC(=O)NCC2CC2)CN(C(=O)Nc2cnccc2C(F)(F)F)CC(F)(F)C1 Cc1ccc2c(c1)SC(C(N1CCCC(N(C(=O)C=C3CCCC3)C)C1)=O)C2 N1(C(C2(C3N(C(c4c(CC)non4)=O)CCC3)CC2)=O)CCC(N(C)C)C(C)C1 N1(C(CN(C(C(CC)C)=O)CC(C)(C)N(C)C)=O)CCC(F)(CO)CC1 C1(NC(c2cc(SC)oc2)=O)CC(O)CN(C(=O)CCc2ccc(F)cc2Cl)C1 c1(C(=O)NCC(N2C(CNC(C3(CC)CCCO3)=O)CCC2)=O)ccccc1Cl Cc1cc(C(N2CC(N(C)C(c3cc(Cl)cs3)=O)C(O)C2)=O)nnc1C C1(c2cnn3c(OCC)cc(C)nc32)NC(=S)N(C)C2=C1C(=O)NC21CCOC1 C1(N(C(=O)CCc2cnco2)CC)CCN(C(=O)Cc2cc(C(C)C)on2)C1 c1(C(=O)NCC(C2CCCN2C(=O)C(O)C2CCC2)(C)C)cnn2ccccc12 N1(C(COCC=C)=O)CCC(CCNC(c2cc(C(F)F)nn2C)=O)C(F)(F)C1 C1(C(=O)NCC(CC)N(C)C(c2ccncn2)=O)CC(=O)NC(CC)C1 c1(CC)cc(C(=O)N(C)CCOCCNC(=O)CC2CN(C)CC2O)cc(N)c1 CC1CCN(C(c2cccc(CO)n2)=O)C1CNC(=O)C(N)=O c1(C(N2CCN(C3CCOC3)CC2)C(=O)NCC=C)noc2c1CCC2 N1(C(C2CC(C#C)(O)C2)=O)C(CNC(c2ccnc(CC)n2)=O)CC2CCCC12 N1(C(C(C)(C)SC)=O)CCCC(CCNC(=O)C(C)n2cncn2)C1 CN1CCC(C)(C(=O)NCC(C)(C)NC(=O)CC2(C#N)CC2)C1=O N1(C(C(c2ccc(C)cc2)=O)=O)Cc2ccccc2C1C(=O)NCC1CCCC1 c1(CC(=O)NCCN(C(C(C)OCc2ccccc2)=O)C)c(Br)cnn1C N1(C(CC2C(C)=NNC2=O)=O)CCC2(CCCN2C(c2csc(C)c2)=O)C1 C(=O)(C(C)(C)C)O.CC(F)(F)F.OC c1(C(N2CCC(C(=O)NCC3(CO)COC3)C(O)C2)=O)c(Cl)ccc(Br)c1Cl C1(CNC(=O)CCc2cn[nH]c2)CCCC1NC(C1CCCC1)=O c1(N2CCC(SC(CCC)C(=O)OCC)C2)ncnc2c1ncn2C(C)(C)CO C1(C(N2C(C)CC(NC(C(C3CCCC3)OCC)=O)C2)=O)Cc2cccnc2C1 c1(C(=O)NCC2(CCOC)CC2)cc(CNC(C2CCCS2)=O)no1 C(C)(C)(CC(C)(C)O)NC(C)=O.CCCC(C(=O)N)N(C(=O)CN(C(=O)C(C)C)C)C C(=O)(C(F)CCC(C)C)N1CCN(C(c2cc(OC)ncn2)=O)CC1C CC1CCCC(C(N2CCC(NC(c3cn(C)nc3C(F)F)=O)C(F)C2)=O)CC1 c1(OC2CCCC(C)C2)ccc(Br)cc1C(=O)OCCN(c1ccccc1I)C N1(C(c2ccc(SC)s2)=O)CCC(C)C(NC(=O)C=Cc2cocn2)C1 C1(CC=C)(NC(c2nccs2)=O)CN(C(=O)C(O)Cc2ccccc2)C1 N1(C(CN2CC(=O)N(C)C2=O)=O)CCC2(CCC2)C(CNC(C2CCOC2)=O)C1 C=CCCC(C(=O)N1CCC(OCC)C1)NC(c1ccnc(O)c1F)=O c1(C(=O)NC(CCCCNC(c2ccnc(OC)n2)=O)C)cc(O)nc(O)c1 C1(NC(c2cc[nH]n2)=O)(CF)CCN(C(C2(c3cnn(C)c3)CCCO2)=O)C1 C1(C)(CNC(C(n2ccc(C(F)(F)F)n2)C)=O)CCCN(C(=O)C=CCF)C1 c1(C(=O)NCC2C(NC(c3ncc(OC)cn3)=O)CC2)c[nH]c2cc(O)ccc12 c1(C(=O)NC(C2(O)CCN(C(=O)C(C)CO)C2)C)c[nH]c2cccnc12 c1(CC(N2C3CN(C(C4(N=[N+]=[N-])CC4)=O)CC2CC3)=O)cccc2ccccc12 C1(CC(=O)OC)CCCN(C(=O)CC=CCNC(=O)C=CC(F)(F)F)C1 C1(NC(C(CO)N(C)C)=O)(CO)CCN(C(c2conc2C(F)(F)F)=O)CC1 N1(C(c2nn(C)cc2Br)C(=O)NCC(C)C)Cc2ccccc2C(CO)C1 C1(F)(CC(=O)NC2C(CCOC)CCC2)CCN(C(C2C3CCCCC23)=O)C1 N1(C(C(C(=O)N(C)C)(C)C)=O)C2CCCC1CN(C(C1(C)CCCCO1)=O)C2 CCCC(CNC(C1CC(N(C)C)C1)=O)NC(c1cc(OC)ns1)=O C1(C(=O)OC)CCC(O)CN1C(c1nccnc1OC)C(=O)NCCOC1CC1 N1(C(CCC=C(C)C)=O)CC(C(N2CC(N3CC(C)(C)C3)C2)=O)C(F)C1 C1(CC)CCN(C(c2ccc(OC)o2)=O)C1CNC(=O)COc1ccccc1 C1(NC(c2ccn(CCCC)n2)=O)COCCN(C(=O)CC2C=CS(=O)(=O)C2)C1 N1(C(C2CCC(=O)O2)=O)CCC2CCCC12C(N1CC2(C=CCO2)C1)=O CCC(CC(=O)NC1CCCC1CNC(c1cc(C)nn1C(F)F)=O)C1CCC1 C(=O)(CCC(F)(F)F)NC(COC)CNC(C1CCN1C)=O C1(C)(CNC(C(=Cc2ccccn2)C)=O)COCCN(C(c2csc(C)c2)=O)C1 Cc1cc(F)cc(C)c1C(N1CC2CC1CN2C(c1ncc[nH]1)=O)=O N1(C(c2cc(COC)no2)=O)CCCC(Cc2ccc(OC(F)(F)F)cc2)C1 CCCC(CCCNC(=O)CCc1cc(C)[nH]n1)NC(c1ccc(CO)cc1)=O C=CC1(C(=O)N(c2ccc(O)cc2C)C)CCN(C(C2CNC(=O)O2)=O)C1 N1(C(C2C(OC)CC2)=O)CC2(CCN(C(C3(C4(O)CCOCC4)CC3)=O)CC2)C1 CC1C(C)CCN1C(C1(CCNC(=O)C=CCO)CC1)=O N1(CC(=O)NC)CCOC(C)(CNC(C2CCCCN2C(=O)C(C)C)=O)C1 c1(C(=O)NCC2(NC(c3c(C)nn(CC(F)F)c3)=O)CC2)cnc2[nH]cnc2c1 CC1CN2CCN1C(C(N1CCCOC(CNC(c3cc(CF)on3)=O)C1)=O)C2 N1(C(C2(c3ccsc3)CC2)=O)CCCC1CCNC(C1(C(=O)NC2CC2)CC1)=O CC(C)CCC=CC(N1CCC(CNC(c2coc(Cl)n2)=O)C1)=O c1(CC(=O)NCCN(CCC)C(C2CC23CCC3)=O)ccc(OC)c(OC)c1Cl C1(C(N2CCCC(NC(C3C(C#C)C3)=O)C2)=O)COc2ccc(OC)cc2C1 C1(C2CCN(C(C3CCCNC3=O)=O)C2)(NC(C(CCC)O)=O)CC1 Cc1cc(C2CC2)ccc1NC(C1CCC(C2CCNCC2)O1)=O C#Cc1cncc(C(=O)NCC2CCCN2C(=O)C(CC)NC(c2ccco2)=O)c1 C(=O)(C(C)CC(C)(C)C)N(CCNC(C1(C(C)C)CCC1)=O)CC1CCCCC1 C1(NC(CCC(=O)NCC)=O)CC12CCN(C(C1CC13CCCCCC3)=O)CC2 CC1(C)C=CC(NC(=O)Nc2nc(C3CC3)cnc2Br)CC1 C(=O)(CCCC(=O)NC(C)CCCCNC(=O)C(C)n1ccnc1)NC(C)C C1(CCN(C(=O)C(=O)NCC2CC2)C)CCCCN1C(=O)CC(F)(F)F C1(C(=O)NC(C2CCCC2)CC)CC2(CC2)CN1C(=O)C1=CCCSC1 c1(C(=O)NC2CN(C(C(C)OCC)=O)CC2C)cc2c(Cl)c(Cl)ccc2[nH]1 CC1CC(NC(c2ccnc(N(C)C)c2)=O)CN(C(=O)CCCC2CCCC2)C1 C1(C(=O)Nc2c(SC)cccn2)COC2(C1)CN(C(=O)Cc1nc[nH]n1)C2 c1(OCC#C)ncccc1C(=O)NC1CCC(NC(=O)C(C2CCC2)OCC)C1 N1(C(c2c(C(C)C)ccs2)=O)CCCCC1CCNC(C1CCCC(=O)O1)=O C(=O)(C(CCC(N)=O)n1cc(CCO)nn1)N1CCSC(C)C1C N1(C(CC2ON=C(CC)C2)=O)CC(NC(c2c[nH]nc2C)=O)C2(CCC2)C1 c1(C(N2CC(C)C(NC(c3ccc([N+](=O)[O-])[nH]3)=O)C2)=O)ccc2c(c1)CN(C)C2 C=CC1(C(=O)NCC2(NC(=O)C=CBr)CCC2)CCC1 C1(CNC(C2C(C)(O)CCC2)=O)CCCC2(CN(c3nc(C#N)c(Cl)s3)C2)O1 N1(CCC)CCCC1C(=O)NCc1nc(C(=O)NC(c2nncs2)C)co1 c1(C(CC)C(=O)N2CCCC2C(C)NC(=O)Cn2cnnn2)ccc(OC)cc1 C=CC(C)(CC)C(=O)NC1COCCN(C(=O)CCCCF)C1 N1(C(C(CC)(C)OC)=O)CC2(C1)CN(C(=O)CCc1cnc(C)s1)C2 C1(NC(CCOCC(C)(C)C)=O)CCCCCC1C(=O)NC1CCC(CO)CC1 c1(C(N2C3C(NC(c4c(C)cnn4C)=O)CC(C3)C2)=O)[nH]cc2c1CCCC2 C(=O)(CS(=O)CCC(F)(F)F)NC1C=CCN(C(c2c(N)cc(F)c(F)c2)=O)C1 C1(NC(Cc2c(SC)cccc2)=O)CCN(C(=O)Cc2ccco2)CC12CCC2 C=CCC(C)(CC)C(=O)NCC(C(=O)NCCC(=O)OC)OC C1(C(=O)NCCOCCCN(C)C(C2CCS(=O)CC2)=O)CC(F)C(=O)N1 c1(NC(c2ccc(CC(=O)OC)cc2)=O)c(N=O)cnn1C N1(C(CN(C2CCSC2)C)=O)CCC(CO)(CNC(=O)CCC2CC2)CC1 C1(NC(=O)Cc2cnns2)CN(C(=O)C=CSc2ccccc2)CC1C1CC1 O=C(CC1COCc2ccccc21)NC12CC(NC(c3cc(O)cs3)=O)(C1)C2 N1(C(c2nc(OCC)sn2)=O)CCN(C(=O)C(=Cc2ccccn2)C)CC1C C(CN=c1cccc(S(=O)(=O)NC2CC2c2ccn(C)n2)[nH]1)c1nnc(C)s1 C1(Nc2nc(C)nc(Cl)c2)CC2(CCC(NC(C3(C(C)(F)F)CC3)=O)CC2)C1 c1(-c2c(C)occ2)nc(CCC2CCOC2)n(-c2ccccc2)n1 CC1(C)OC(C(N2CCN(C(=O)CC3CC(F)(F)C3)C(CF)C2)=O)C(C)(C)O1 n1(CCC)ccc(C(=O)NC2(CNC(=O)CCCNC(N)=O)CCC2)n1 c1(C(C)NC(=O)CC=CCNC(=O)CCC2CCCO2)nnnn1C c1(C(N2C(CNC(c3cccc(OC)c3)=O)CCC2)=O)c(C)nn(C2CC2)c1Cl C12(NC(CCc3ccc(C)s3)=O)CCCC1CN(C(=O)C(F)(F)C1CC1)C2 C1(O)(CNC(CC2CC(CC)C2)=O)CCCN(C(=O)CCN2CCCC2=O)CC1 C1(C(=O)NCCC(=O)OCCc2cnn(C)c2)(OCC)CCCCC1 N1(C(C2C(C)CCOC2)=O)C(C(=O)NCC(CO)C2CCC2)CCC12CC2 C1(CC(=O)NCCN(C(C2COCCO2)=O)CC2CC2)CC2(COC2)C1 CN1CCN(C(N2CCC(C(=O)Nc3ncccc3Cl)CC2)=O)C2CC12 C1(NC(C2(CC)CC2)=O)CCCC2CN(C(c3cc(O)ccc3O)=O)CC12 N1(C(C=CC(C)C)=O)CCN(C(c2nc(C(F)(F)F)cs2)=O)C2(CC2)C1 c1(C(N2CC(CNC(CN(CC)CC)=O)C2)=O)ccc(O)c(CO)c1 Cc1cc(C(C)(C)C(=O)NC(C)CC(C)NC(=O)Cc2ccsn2)cs1 c1(C(=O)NCC(CNC(C(CCC#C)O)=O)OC)cc2c(C)cccn2n1 N1(C(c2c(OC)scc2)=O)CC(C(=O)NC2(C(C)O)CC2)CC(C)C1 c1(NCC(=O)NCC(c2ccccc2)CNC(C(F)OC)=O)n[nH]c(O)n1 N1(C(C=C(CC)CC)=O)CCCC(C)(CNC(C2(OC)CCCOC2)=O)C1 C(=O)(C(CC(C)(C)C)OC)N1CC(O)(CNC(C2C(=C)C2)=O)C1 c1(OC)ccc(Cl)c(C(=O)NCC(C)(CC(C)C)NC(C2CC(O)CN2C)=O)n1 C(=O)(C1=COCC1)N(CCC(C)Br)C(C)(C)C C1(CNC(c2cc(CC)n(C)n2)=O)CC2(CO1)CN(C(C1(C)CC(C)(C)C1)=O)C2 C(C(C)CC(=O)N1CCSCC1CCNC(=O)COC1CC(F)(F)C1)OC N1(C(=O)Cc2ccc(F)cc2)CCCC2C1CCN2C(c1ccc(F)cc1Cl)=O CCC(C#N)(CC)C(=O)NCC1CC(CNC(=O)C(C)(Cl)Cl)CO1 CCCC(CC(=O)NCCCC1CC1)NC(c1cncnc1)=O C1(C(=O)NCCC2CN(C(C3SCCCS3)=O)C2)CCC(F)(F)CC1 N1(C(c2nc(C)c(-c3ccc(N(C)C)cc3)cc2)=O)CC2CCC(C1)N2C CC12CCCC(C(N3CCOC(CNC(=O)Cc4nccs4)C3)=O)(CO1)C2 c1(OCC)cc(Br)c(F)cc1NC(C1C=CC(NCc2ccc(COC)o2)C1)=O C1(OC)CC(CNC(=O)Cc2csnn2)N(C(c2cn(CC(F)F)nc2C)=O)C1 CC1CCc2n[nH]cc2C1C(=O)NCc1cccc(NC(=O)CC(=O)NC2CC2)c1 N1(C(C=CCC(C)(C)NC(CC(C)F)=O)=O)CCC2(CNC(=O)N2)C1 N1(C(C2C(CC)C2)=O)CCC2CN(C(C3COC(=O)O3)=O)CC2CC1 C1(C)(CNC(CCC2CCC(NC(CC3CC(=C)C3)=O)C2)=O)C=CCCC1 c1(C(=O)NC(C)CNC(C2CCCC2CF)=O)cccc(-c2ccco2)c1 C1(C(N2CC(C)CC2)=O)CC=CCC1C(=O)Nc1ccc(NC(C)=O)cc1.CO c1(C(=O)OC)nc(=NCC2CCC(NC(c3cnoc3C(C)C)=O)C2)cc[nH]1 c1(OC)nc(C(=O)NC2CC(C)(NC(c3cncc(F)c3)=O)C2)sc1C n1(CC(N2CCC(N(C(=O)C=C3CC3)CCC)CC2)=O)nc(C)ccc1=O N1(C(CCCC#CC)=O)CC(NC(c2cnc(C(F)F)s2)=O)C2(CCOCC2)C1 CC1CCC(NC(=O)CC=C(Cl)Cl)CN1C(=O)Cc1ccc(-c2nnco2)cc1 C1(CCNC(C2C(C(C)(C)C)CC2)=O)COCCN1C(c1cc(C(N)=O)co1)=O c1(CN(C(CNC(C(C(C)C)NC(N)=O)=O)C)C)cc(O)nc(O)n1 c1(C(=O)NCCC2(NC(c3cccc(C)n3)=O)CC2)nccc2ccsc12 Cc1nscc1C(=O)N(CC(C)NC(C1CC1F)=O)C Cc1cccc(C(=O)NC2CCC(C)(CNC(c3cccc(O)n3)=O)C2)c1C c1(CC)ccc2occ(C(=O)NC3CN(c4cc(C)nc(C)n4)CCC3C)c2c1 Cc1cc(C(=O)NC2CCCC(NC(C3CC(C)(O)C3)=O)C2)cc2cccnc12 C12(CNC(C=CCC)=O)CC(COC)(CN1C(=O)CC1CCCCC1F)C2 N1(C(=O)Nc2c(C)ncc([N+](=O)[O-])c2)CCC2(CC1)CN(c1nnco1)CCO2 c1(CC(=O)NCC2C(NC(c3c(SC)scc3)=O)CC2)ccc([N+](=O)[O-])cc1 C1(CNC(C(=O)NCCc2scc(C(C)C)n2)=O)CCC2(CC2)C1 Cc1cc(Cl)ccc1-n1nc(CCn2cccc2)nc1CC(F)(F)F C(=O)(C(C)CC(C)C)NC(c1c(CC)cccc1)CNC(=O)CC1CC1 c1(NC(N(C)Cc2ccc(OC)c(Br)c2)=O)ccc(C2=CCCCC2)cn1 N1(c2ccc(CC)c(F)c2)C(=O)NC2(CCC(F)(F)CC2)C1=O Cc1ccc(CN2CCCC(NC(=O)CCc3cccc(F)c3F)C2)c(F)c1 N#Cc1ccc(Br)c(NCC2(N3CCNCC3)CCOCC2)c1F C(=O)(n1c(=O)c(C#N)nnc1S(=O)(=O)c1cccnc1)C1(C)CC1.o1[nH]c(=O)o1 c1(C(N(CCCN(C)C(c2ccnn2C)=O)C)=O)ccc2c(c1)CC(C)(C)O2 C[Si]1(C)CCC(NC(=O)NCc2ccc(C(F)(F)F)cc2)CC1 c1(CN(C(C(C)=C2CC2)=O)C)cccc(CNC(c2ocnc2C)=O)c1 C(C)(C)(CCC(=O)N1CCC(C)C1C(N1CC(S(C)=O)C1)=O)OC c1(CNC(C2CC(NC(COCCC=C)=O)C2)=O)ncc(CO)[nH]1 Cc1cccc2[nH]cc(CCNC(=O)C(C3CCC(F)(F)CC3)O)c12 CCCCC(CNC(=O)COc1ccsc1Cl)NC(C1(CO)CCC1)=O C(=O)(CCCCCC(C)O)N1CCCC(CNC(CSCCOC)=O)(OC)C1 c1(CC)ccc(CC(=O)NC2CCN(C(C3COCCN3C)=O)C2(C)C)cc1F c1(C(=O)NC2CC3CN(C(CC(=O)OC)=O)CC32)ccc2oc(C)nc2c1 CCCC(CCCO)C(=O)NCC1CC2COCC2N1C(=O)C(C)NS(C)(=O)=O C1(C(=O)NCc2nccc(OC)c2)CN(C(=O)CC2CC=CCN2C)CCC1(C)C C(=O)(C1=CCCCCC1)NCC(CN(C(=O)CC1(n2cncn2)CC1)C)O C1(C)(CC(=O)NCC(C)CN(C)C(c2cscc2Br)=O)CC(F)(F)C1 c1(C(N2CCC(NC(CC3(C=C)CCC3)=O)C23CC3)=O)ccc2c(c1)OCCO2 c1(C(=O)NC2CCC(C(N3C(COC)CCCC3)=O)CC2)c(C)cnnc1O c1(C(=O)NCCCN(C(C(C(C=C)C)C)=O)C(C)C)cc(S(N)(=O)=O)ccc1C C1(C(=O)NC2CC(CCNC(c3sccc3OC(F)F)=O)C2)CC2C=CC1CC2 C1(NC(CSc2ccccc2)=O)CCC2(CCC2)CC1.O=c1c(=O)[nH]1.C1C(=O)N1 C1(C)(C(N(C)Cc2ccc(OC)c(C(F)(F)F)c2)=O)CCOC2(CCC2)C1 c1(NC2CCC(C[N+](=O)CN3CCCC3)C2)ncnc2ccccc12 N1(C(CC2N(CC)CCOC2)=O)CCN(C(C2CNC(=O)N2)=O)C(CCO)C1 c1(NC(C2CCC(CCNc3ncncc3Br)CC2)=O)cc(F)cc(F)c1 C1(N(C(CC)C(C)C)C(C(=O)C(F)(F)F)=O)CCC2CCCCC2C1 Cc1cccc2cc(C(N3CCC(O)C(NC(=O)C(F)(F)C(F)(F)F)C3)=O)[nH]c12 C(C(C(=O)N1CCCCC1CNC(=O)CS(=O)(=O)N(C)C)C(F)(F)F)OC CC(C)(C)CC(O)CC(=O)N1CCC12CN(C(=O)C(CCO)c1ccccc1)C2 C1(O)(CNC(CCCOCCC)=O)CCCN(C(=O)Cc2csc(C(C)C)n2)C1 n1(CCC(N2C3CC(NC(=O)COC(F)F)C(C3)C2)=O)ncc2ccccc12 N1(C(=O)NC2CCOCC2C(=O)O)CC2CC1(Cc1ccccc1)CO2 Cc1cc(C(=O)NCC(C2CCC2)NC(=O)C(=O)C(C)(C)C)ncc1CO C1(NC(c2cc(C)no2)=O)CC2CN(C(=O)COCCCC(C)C)CC2C1 C1(C(=O)NC(C(C)C)CCN(C(=O)C(C)NS(C)(=O)=O)C)CCCC2(CCC2)C1 N1(Cc2c(C)non2)CCC(NC(=O)CCn2cccnc2=O)C(C)C1 c1(OC)ncc(C(N2CC(C)(OCC(=O)NCCCC3COCC3O)C2)=O)cn1 C1(NC(=O)C=CCF)CN(C(c2ccnc(S)c2)=O)C2(CCCCCC2)C1 c1(NC(C2OCCN(C(C3CCC(C)O3)=O)C2)=O)ccc2ncccc2c1C#N N1(C(=O)OC)CCOC(Cc2cn(CC(=O)NCC3(CC4CCC4)CC3)nn2)C1 C1(CNC(C(C2CC2)OC)=O)CC(F)CN1C(=O)C(C)CCO C1(NC(CCN(C(C(c2cncnc2)C)=O)CCO)=O)CCN(C)C(=O)C1 C1(C(=O)NC(C(=O)OCCC)C)CC12CC(NC(c1ccncc1F)=O)C2 C=C(C)C1OCCC1C(=O)NC1(C(=O)NOCCC(C)O)CC1(C)C C1(CC(N2CC(C)(NC(c3c(CC)nco3)=O)C2)=O)CC(c2ccccc2)=NO1 c1(C(=O)NC2CC(NC(Cn3c(C)c(Cl)cn3)=O)C2)cccc2c1OCCN2C C1(C(=O)NC2CCC(NC(=O)CCCN3CCCC3)C2)C2CCC(F)C12 C(=O)(CCS(=O)(=O)C1CCCC1)NC1CC(NC(CC2C(C)(C)C(O)C2)=O)C1 N1(C(CCC=C)=O)CCCC(C2CN(C(c3cccc(S(C)(=O)=O)c3)=O)C2)C1 C(CCN=C(NCCNC(c1ccccc1)=O)N1CCC(C2CCOC2)C1)OC N1(C(CN(C(c2cn(C3CC3)nn2)=O)CC)=O)CCC(OCC(C)C)CC1 N1(C(C(C=C)O)=O)CCCC(n2cc(-c3ncc(F)cn3)nn2)CC1 c1(C(N(C2C(C)CN(C(C3CSC3)=O)CC2)C)=O)ccn2c(O)nnc2c1 C(=O)(C(C1=NOC2C3CCC(C3)C12)N1CC(F)CC1C)NCCCSCC N1(C(C(CC)n2ccnc2)=O)CC(C(=O)N(C)Cc2cnc(C)cn2)C(C)(C)C1 n1(CC(=O)NCC2C(NC(C=CC(CC)=CC)=O)CC2)ncc(C)cc1=O C(N=c1cccc(S(=O)(=O)N2CCCC2CCC)[nH]1)C1(CCC)CC1 C(C(N=[N+]=[N-])C(=O)N1CC(C(=O)NC2CN(C(=O)NCC(C)C)C2)(SC)C1)CC C1(NC(C2C3CCCC23)=O)CN(C(C2(Cc3ccccc3)CC2)=O)CC1F C1(C(N(C)Cc2ccsc2)=O)CCCN1C(c1cc(Cl)cs1)=O C(=O)(C(C)C(C)S(C)(=O)=O)NC1CCN(C(c2ccc(CC)c(Cl)c2)=O)CC1C Cc1c(Br)ccc(F)c1C(N1CCCC(NC(c2cnc3ccccn23)=O)C1)=O Cc1cnc(NC(C2CCN2C(C2(C)CC2)=O)=O)s1 N#CC1CN(C(=O)C(=O)Nc2ccnc(OCC(F)(F)F)c2)CC1O c1(N(C)CC2CCC(F)(F)CC2)nc2c(c(=NC3CCC(CO)CC3)[nH]1)SCC2 C(=O)(C(C)(C)CCSC)N1CC2C(NC(CCOCC(C)C)=O)(C2)C1 C1(C(=O)NCC2N(C(c3c(C)oc(CO)c3)=O)CCC2)CCC2(CC1)CC(O)C2 c1(C(=O)NCC2C(NC(=O)COCc3nc[nH]n3)C2)cc(-n2cccc2)[nH]n1 c1(C(N2CC(C)CC2c2cccc(OC)c2)C(=O)NC)cc(Cl)c(F)cc1F N1(C(CC=CCC)=O)CC2CCCC2(CNC(c2ccc(C#N)cc2)=O)C1 CCC(N=c1[nH]c(=NCC2(C)CCCCC2(C)C)[nH]c2cccc(F)c12)C1CC1 C=CC1(C(=O)NCC2CCCC2N(C)C)CCN(C(=O)CC2CCCCCC2)C1 C(CO)(CCCCNC(=O)CCCC(C)=O)NC(Cc1c(CC)cccc1)=O c1(C(C(=O)NC2C(NC(c3n(CCC)ccc3)=O)C2)C2CC2)ccc(F)cc1 N1(C(c2cc(C)no2)=O)CCC(CCNC(=O)Cc2cc(C)ns2)CC1C c1(C(=O)NC(C(C)C)CCNC(=O)CC(C)c2ccco2)ccn(C)c(=O)c1 C(C)(C(C)(C)C(=O)NCC1(C2CC2)CCCO1)NC(C(C)NC(N)=O)=O c1(C(N(C(C)CNC(c2cc(-c3cccs3)on2)=O)CC)=O)cc(C)cs1 C1(CNC(CC(CCC)O)=O)CC2COCC2N1C(C1CCCC(O)C1)=O CC(C)(C)C(C#N)C(=O)N1Cc2[nH]nc(C(=O)NC3(C4CC4)CCOCC3)c2C1 CCCCC(CNC(c1ncccc1OC(C)C)=O)NC(=O)Cc1n[nH]c(C)n1 C(=O)(CCC(F)(F)F)N1CC(C(C)NC(=O)CC2(C)CCCO2)OCC1 c1(C(N(C)CC2CCCCN2C(=O)C(O)C(F)F)=O)cccn2cncc12 c1(OC)nn(C)cc1C(=O)NCC1CCCC1NC(=O)Cn1cc(C#N)cn1 C=C1CC2(C1)CN(C(=O)CC(C)CNC(c1cc(C)c(CC)o1)=O)C2 c1(C(N(CC(C)NC(CC2(OCC)CCC2)=O)CC)=O)occc1C1CC1 c1(OC)cc(CN2CC3CC2CN3c2ncc(F)cn2)ccc1O c1(CC(N2CCC(C(C)NC(c3c(C)nc(O)[nH]3)=O)C2)=O)cc(F)ccc1F C1(C(C)C)(CO)CCN(C(=O)CC(C)NC(C2CC3(CSC3)C2)=O)C1 N1(C(Cc2ccc(C)nc2)=O)CC(NC(=O)C(c2ccccc2)F)C2(CC2)C1 C1(C(=O)NC(C)CCN(C(=O)C(O)CC2CC2)C)CCC(C)CC1 C1(C)(C(N2CC(C(C)NC(C3CCOC3)=O)C2)=O)C=CCC1 CCC(C)CC(C)NC(C1(NC(C2CC(CC3CC3)C2)=O)CC(F)(F)C1)=O c1(C(=O)NCC(CC(F)(F)F)NC(C2(CCC=C)CC2)=O)cc2n(c1)CCCC2 C1(NC(Cn2c(C(C)C)nnn2)=O)CN(C(=O)CSCCC#N)C2CC12 c1(C(=O)NCC2(CO)CCN(C(CCS(C)=O)=O)CC2)cnc2ccoc2c1 c1(-c2cccc(SC)c2)ccc2c(CC(=O)Nc3cc(F)ncc3F)n[nH]c2c1 C(=O)(C(O)C(C)CC)NCc1c(C(=O)NC(N2CCCCCC2)CC)cccn1 N1(C(C2(C(=O)OC)CC2)=O)CCC(C)C1.c1(CNC=O)cccc(-c2ccoc2)c1 c1(C(=O)NC2(CNC(c3c(SC)cccc3)=O)COC2)c(O)c(Cl)cc(Cl)c1Cl c1(CC(=O)NCCC2CCNC2)ccc(NS(N)(=O)=O)cc1 CCCC(F)C(=O)NCC(CC(=O)NC(C)(CC)CO)C1CCC1 C(=O)(CC(O)CNC(c1c(C)noc1C)=O)NC(c1ccn(C)n1)CC C1(F)(CNC(Cc2ccc(OC)cn2)=O)CCN(C(c2cc(F)c[nH]2)=O)CC1 C#CC1(NC(=O)C(O)CNC(c2cc(C)nn2C)=O)CC2CCCC12 N1(C(C(CC(C)C)NC(N)=O)=O)CCC2CN(C(=O)CC3CCCCC3)CC12 CC(CC1CCC1)C(=O)NC1CC(CNC(c2c[nH]nc2C(C)(C)C)=O)C1 C1(CC#C)(NC(=O)C(C2CCN(C(c3ccc(Cl)o3)=O)C2)F)CC=CCC1 N1(C(C(C)NC(N)=O)=O)CCC(CNC(C2(c3nncs3)CC2)=O)C(C2CC2)C1 N(C1CN(C(=O)Cc2cccnc2F)Cc2ccccc21)C(C(C)C(C)(C)C)=O C1(N(C(=O)Cc2cc(-c3ccco3)on2)C)CCC(NC(C2(C#N)CC2)=O)CC1 c1(C(=O)NCC(CCOC)NC(C(C=C)C)=O)cccc2occc12 c1(C(CC)C(=O)N(CC(CC)NC(=O)Cc2cnn(CC)c2)C)c(C)noc1C C(CCN=c1[nH]nc(C(N)=O)s1)OCCNC(C1CCCN(C)C1)=O C1(COC)CC(CNC(=O)CN2CCC(C)C2)N(C(c2cnc(O)n2C)=O)C1 S(=O)(=O)(CCCS(=O)(=O)N(c1ccncc1C(F)F)C1CC1)NC(C)(C)C#N C1(NC(Cc2cc(C)[nH]n2)=O)CN(C(=O)CC(c2c(C)n[nH]c2C)C)CC1O C1(CC(=O)NCCCN(C(=O)C=CC2CCC2)CC)CCCC(C2CC2)O1 c1(C2(N(C(=O)C(C)CF)CCCCC3CN(C(C)=O)C3)CC2)ncc(Cl)cn1 C1(OC)CC(CCNC(=O)CC2C=NN(C)C2=O)N(C(c2cc(CO)on2)=O)C1 C1(CC)CN(C(=O)C(C(C)C)NC(=O)C(C)C)CCN1Cc1cc(C)on1 N1(C(C2(S(C)(=O)=O)CC2)=O)CC(NC(c2nncs2)=O)C2(CCOCC2)C1 N1(C(C2CCN(CC(C)C)CC2)=O)CCCC(O)(CNC(=O)CN2CCC2C)C1 c1(C(=O)OC)ccc(C(=O)NCC(CO)NC(C2CCC2)=O)c(Cl)c1 c1(C(=O)NC2CCN(C(c3cc(OCC)n[nH]3)=O)C2C)cnn2ccc(O)nc12 C1(NC(=O)COC2CCOC2)CC2CCC(C1)N2C(c1csc2cncn12)=O Cc1cc(C)c(C(N2CCCC(NC(=O)C3=CSCS3)C2)=O)cn1 C(C(C)(C)C(=O)N1CCC(C(C)C)C1)N(C(C(CC)=CCCC)=O)C c1(C(C(N2CC(=C(CNC(CN3C(C)CC3)=O)F)C2)=O)C)ccn(C)n1 CC1NC(=O)CCC1NC(=O)Nc1ccc(N2CCN(C(=O)C3CC3)CC2)nc1 Cc1cc(O)ccc1C(N1CCN(C(c2occc2F)=O)CC1C)=O c1(C(=O)NC2CCN(C(C=CC(C)(C)SC)=O)CC2O)cncc2n[nH]cc12 c1(OC)cn(CC(N2CCCC2CNC(c2cc(Cl)sc2Cl)=O)=O)c(C)cc1=O N1(C(C=CCOC)=O)CC2(CCN(C(=O)C=CCOC)CC2)C2COCC12 C(CCC(C)(C)NC(=O)C(CC)NC(C)=O)NC(C(C)OCCCC)=O C1(CNC(C2(SC)CC2)=O)C2CN(C(C3(C)CCCO3)=O)CC12 c1(-n2cc(NC(CC)C(=O)OC)nn2)cccc(-n2cnnn2)c1 c1(C(N2CCC(CC)CC2)C(=O)Nc2ccccc2)cnc2cc(C)nn2c1 c1(CC(=O)NCCC2(CNC(C(CCC)OC)=O)CC2)ccc2c(c1)NC(=O)C2 C1(C(=O)NCC(=O)Nc2nnc(O)nc2O)CN(C(=O)C(F)OC(F)(F)F)CC1(F)F C1(N(C(=O)CN2CCCC2C)CC)CCN(C(=O)C(C)(CC)OC)CC1 C1(C(N2CC(CC(=O)NCC3(C=C)CCC3)(OC)C2)=O)CC12CCCC2 c1(C(=O)NCC2(C(=O)NC(C)C(O)C(F)F)CC(=C)C2)cc(C)c(C)o1 N1(C(C=CC)=O)CCN(C(=O)C=Cc2ccsc2Br)CC1CS(C)(=O)=O C1(OC)CN(C(c2cncn2C)=O)CCC1NC(=O)C#CC(C)(C)C C1(CNC(=O)OCC)CN(C(C2(CC(C)C)CCC2)=O)CC2(CCC2)O1 C#Cc1cnn(C)c1C(=O)NCC1CN(C(=O)CC2CC(F)(F)C2)CC1(C)C c1(C(N2CCC(N(C(CNC(CC)=O)=O)C)C2)=O)cc(S(N)(=O)=O)co1 c1(C(=O)NCC2CC(CNc3c(C#N)cccn3)OC2)ccnc2[nH]nnc12 N1(C(c2ccc(CC)o2)=O)CC(NC(c2ccc(C#N)s2)=O)C(C)C1 N1(C(CC2(OC)CN(C(CNC(=O)NC)=O)C2)=O)CC2CCC(C(N)=O)(C2)C1 C=CC1(C(=O)O)CCN(C(=O)C(C)(C)C)CC1 CCC(C(=O)N(C)CC=CC(=O)N(C1CCCC1)CC)C(C)(C)CC C1(C(=O)NCCSC)COC2CN(C(c3ccc(I)cc3)=O)CC12 C(C(=O)N1CC2(CCC2NC(=O)CCn2ncn(C)c2=O)C1)(C(C)(C)C)N(C)C C1(NC(C2(c3ccn(C)n3)CC2)=O)(CNC(=O)CCN2CCCC2)CCCCC1 N1(C(c2cnc(CC)s2)=O)CCCC2(NC(=O)C=Cc3cc(C)no3)CCCC12 C(=O)(CC(CNC(=O)C(C)=CCCSC)C1CCC1)NC(c1ccccc1)C#C c1(N(C(C(=O)NCCCF)C2C(CC)C2)C)ccccn1 N1(C(CCCCOCCC=C)=O)CCCN(C(=O)CC(C)(C)C(=O)OC)CC1C N1(C(CN(CCC)C)=O)CCc2ccccc2C1CNC(c1cc(C)[nH]c1C)=O c1(C(=O)NC23CCC(CNC(C(CCC)O)=O)(OC2)C3)cc(C)c2c(c1)CCC2 N1(C(C(C)C2CCC2)=O)CCC(C2CCN(C(=O)CNS(=O)(=O)N(C)C)C2)CC1 c1(OC)cc(C)ccc1OCC(=O)N(CC(O)CNC(=O)Cc1csnn1)C C1(C(N2CCN(C(CCSCC)=O)C(COC)C2)=O)CCc2cnnn2C1 Cc1[nH]c2ccc(F)cc2c1CC(=O)NCCN(C)C(C1(F)CCCOC1)=O c1(C(N2CCC(OC)(CNC(c3cccn3C)=O)C2)=O)ncc2n1CCCC2 C1(CNC(=O)COC2CCN(C(c3cccnc3)=O)C2)CCC=CCC1 C1(C(=O)OC)(C(=O)NCC(O)CCNC(c2ccccc2)=O)C2CCC12 c1(CC)ccc(C(=O)NCC2COCCN2C(c2csc(Cl)c2)=O)cc1[N+](=O)[O-] N1(C(CCc2ccc(OC)cc2)=O)CCC2CCCN(C)C2C1 C(=O)(CC(C(F)(F)F)NC(C1CC2(CCO1)CC2)=O)NC(C)C(C)(C)C#N C1(CC)(CNC(=O)NC(C(C)(C)CO)c2nccn2C)CCCCO1 c1(C(=O)NC(c2cccc(Cl)c2)CNC(C(CC)C#N)=O)c(OC)cccc1F C1(NC(CSCc2cccc(C)c2)=O)CCN(C(=O)C=CC2CCC2)CC1C c1(CCCCNC(=O)C(=O)NCC2CC3C=CC2C3)ccc(Cl)nc1 n1(C(C)C)ncc(F)c1C(=O)NC1CC(CO)N(C(=O)C(C)c2ccco2)C1 C1(C(N(CCOCC)C)=O)CN(C(C2(C)CCCS2)=O)CC12CC2 C(=O)(CCS(C)(=O)=O)NC(C(=O)NCCC1CN(C)C(=O)C1)CCC1CCC1 CC1(CNC(=O)CC(CNC(c2cnc(S)nc2)=O)C2CCC2)CCCC1O N1(C(C2=CCC(NC(C3(CC#C)CCCO3)=O)C2)=O)CC(C)(C)OC(C)(C)C1 c1(C(=O)NCC(C2(O)CCN(C(=O)C#CC3CC3)C2)C)ccc(C2CCC2)nc1 CCCC(C(=O)NCC(C)(O)CNC(c1cn(CC)cn1)=O)C(C)C c1(-c2cc(C(N(C(C)CCNC(=O)CC(C)(C)C)C)=O)no2)ccc(F)cc1F C(=O)(C1=C(C)CC1)NCCOC1CN(C(C(C)(C2CC2)OC(C)=O)=O)C1 N1(C(C(C)NC=O)=O)CCC2CCC(NC(C3COCCN3C=O)=O)C1C2 N1(C(CC2CCCC(CNC(=O)OC(C)(C)C)C2)=O)Cc2cc(O)nnc2C1 C(=O)(C1=C(C(=O)N2CCCC2C(=O)OC)CC1)OC C1(NC(C(C)=CC2CC2)=O)C(C)CN(C(=O)CC2CCC(C(N)=O)CC2)CC1C c1(C(N2CC(CNC(C3CCCN3C=O)=O)CC(C)C2)=O)cc2ccccn2c1 N(C(=NCC1CC1)N1CC(c2ccccc2)C2(CCC2)C1)C(COC)C CCC(O)C(C)C(=O)N(C)CC1CCCN1C(=O)CC1CCC(=O)C1 c1(C(=O)NC(CNC(c2cc(OCC)cc(=O)o2)=O)C)cc(C)cc(OC)c1O C1(CNC(C(C2CN(C(C3CC(F)CN3C)=O)C2)OC)=O)CC(C2CC2)C1 C1(C(N2CC(CC(=O)Nc3cnnc(Cl)c3)OCC2)=O)CCc2ccccc2C1 N1(C(CC)=O)CC2CC3CC2C1C3NC(C1CCOC2(CCCC2)C1)=O C(=O)(CC(C(F)F)NC(=O)C=C(C)c1ccco1)NC(COC(C)=O)CO C1(CNC(c2c(C)occ2)=O)CCC2(CN(CC3CCCC34CC4)C2)O1 C1(NC(COCC(C)C)=O)CC2CN(C(=O)CCc3nnc(O)nc3O)CC2C1 C1(CNC(N(C2CCCC2O)C)=O)CC2OC1C1CC21 C(=O)(CCCC(C)C)N(CCCNC(C(Br)=C(C)C)=O)CCO N1(C(CCS(N)(=O)=O)=O)CC2CC(NC(C3CC(F)C3)=O)C(C2)C1 c1(C(=O)NC2CCN(C(C3CN(C)CC(C)O3)=O)CC2O)cnc2[nH]ncc2c1 C=CC1(CC(N2CC(NC(C3(C(C)C)CC3)=O)C(O)C2)=O)CCCCC1 Cc1ccc(Br)cc1C(N1CC(CCn2cc(CC(O)C3CC3)nn2)C1)=O C1(C(=O)NCc2c(C(=O)NC(c3nnnn3C)C)cccn2)CCCC1C1CC1 c1(C(=O)NC2CCN(C(C3CC(=O)NC(=O)N3)=O)CC2F)cncc2sccc12 c1(SC)cccc(CC(=O)NCCN(C2CCCCC2)C(=O)Cc2cncs2)c1 C=CC1(O)CCN(C(=O)C(CC(F)F)NC(=O)COC2CCCOC2)C1 C12(C(=O)NC3CCN(C(CC4(OC)CC4)=O)C3C)CCCCC(=O)N1CCC2 Cc1nn(CC(=O)NC(CCc2nn[nH]n2)C(=O)O)c(=O)o1 C12(CCNC(C(CC)OC)=O)CCC(C1)N(C(c1cc(C)ccc1OCC)=O)C2 CC1CC(C)(C(N2CC3(CC(NC(c4ccc(N)c(F)n4)=O)C3)C2)=O)CC(C)O1 c1(CC(=O)NC2C(NC(C(CC)(CC)CC)=O)C2)c[nH]c2cccc(F)c12 C(CCCC(=O)NOCC(C)O)N(C(C(C(CC)CC)OC)=O)C CCCCCC(CCCCC)C(=O)N1CC2CN(C(=O)C(C)P(C)(C)=O)CC2C1 C(=O)(CCS(N)(=O)=O)NC1C(C(=O)NCC2(OC)CCC(C)C2)COCC1 c1(C(=O)NC23CC(NC(c4c(C)onc4O)=O)(C2)C3)ccc2cccc(C)c2n1 C1(=CC(=O)NC2C(CNC(C3(OC)CC3)=O)CC2)CCC(C)CC1 CCC(CCCC(=O)N1CCC(CN(C)C)CC1)NC(c1cc(C)cs1)=O c1(C(C(=O)NCC(CC=C)NC(c2nccnc2CC)=O)=O)c(C)nn(C)c1C c1(CC(C(=O)NCC(C=C)O)NC(=O)C(C)SC(C)C)cnn(C)c1O CC1(C2CC2C(N2CC(C3CC3)(C(=O)Nc3ccc(Cl)nc3)C2)=O)COC1 N1(C(C2C(CC)C2)=O)CC(O)CC1C(=O)NCc1nn[nH]c1C1CC1 c1(CC)cc(C(N2CCCC(NC(c3ncc(F)cc3C)=O)C2C)=O)cc(F)c1 N1(C(c2cccc(C)c2C#N)=O)CCC2(CCCC2NC(=O)CCCF)C1 C1(NC(Cc2c(C)n[nH]c2C)=O)CCN(C(c2cccc(O)n2)=O)CC1O C(=O)(C(C)(C(C)C)OC)NCc1cn(CCNC(C2C(C#C)C2(C)C)=O)nn1 C1(CC(=O)NC2(CCNC(CCCCSC)=O)CC2)CC(C)CC(C)(C)C1 c1(NC2CCC(CC)C2)ncc(C)cc1S(=O)(=O)NCCc1cc(Cl)ccc1F CC1(F)CN(C(C2(C3CCC3)CC2)=O)CCN(c2cc(O)nc(=O)n2C2CC2)C1 C1(CC)(CO)CCCN(C(C2CC3(CC(NC(c4ccco4)=O)C3)C2)=O)C1 c1(C(=O)NC(C(=O)NCC2ON=C(C)C2)(C)C)ncnc(O)c1F CC(C)(C(=O)NC1CC(F)CN(C(=O)C(C(C)(C)C)NC(N)=O)C1)C(F)F c1(C(N2C3CN(C(C(CC#C)O)=O)C(C3)C2)=O)coc2c(F)cc(Cl)cc12 c1(OCC(=O)N(C(CNC(c2c(NC)scn2)=O)C)C)ccc(Cl)c(F)c1 c1(C2(CNC(c3cn(C(C)(C)C)nc3)=O)CCC2)ccc(F)cc1 N1(C(C(N2CCOC2=O)C)=O)CCCC(O)(CN(C)C)CC1 c1(C(=O)NCCN(C(C2C(CC)OCC2)=O)CC2CC2)cc(C#N)ccc1Br CC(C)(C)CC(C(=O)NCC(=O)N(C)C)N1CCCC(C)(C(=O)OC(C)(C)C)C1 C1(NC(C=Cc2ccc(SC)s2)=O)CCCCCC1NC(=O)C(C)=C1CCCC1 c1(C(N(C(C)CN(C(=O)C(=O)N(C)C)C)C)=O)ccc2cnsc2c1 N1(C(CC(C)(C)OC)=O)CCC(NC(=O)CC23CCC(CC2)OC3)CC1C c1(C(=O)NC2(CCNC(Cn3nc(C)oc3=O)=O)CC2)nccc2occc12 c1(CNC(Cc2c(C)ccs2)=O)ccccc1CNC(=O)CCC(C)C C1(C(=O)NC2CC(CCNC(CCCC=C)=O)C2)CN=C2N=CNN2C1 Cc1ccc(F)cc1C(=O)NC1(C(N2CCCC(C#N)C2)=O)CC1 c1(C(N(CC(=O)N(CCNC(C)=O)C)CC(C)C)=O)ccc2cncn2c1 N1(C(C23C(C)OC(C)(C2)C3)=O)CC(CO)C2(C1)CN(C(c1nccnc1Cl)=O)C2 C(=O)(CP(=O)(C(C)C)C(C)C)NCC=C1CCN(C(CC(C=C)(C)O)=O)CC1 N1(C(CSCC=C)=O)C2CCC1CN(C(=O)CSCCC#N)C2 C1(CNC(C2CC2CF)=O)CCCCN1C(=O)Cn1nnnc1-c1ccsc1 C=CCCC(=O)N(C)CC1(NC(=O)COC(C)CC)CC1 C(C)(CCCC(=O)NC)NC(CC(C=C)C)c1nn[nH]n1 C(C1C(C(=O)NC2CCN(C(C3COC(=O)N3)=O)C2C)C1(C)C)=C(C)C C(=O)(C1=C(Cl)CCC(C)C1)N1CC(CNC(c2c(C)cc(C#N)cn2)=O)OCC1 CC1(O)CCN(CC(=O)NC23CC2CN(C(=O)Cc2cnccn2)C3)C1 C1(C)(CCC)C(=O)NCCN1C(C1CCC2(CN(CCSC)C2)O1)=O c1(C(c2nnnn2C2CCC2)NCc2nnn(C(C)(C)C)n2)cc(Cl)ccn1 c1(CC)c(C(=O)NCC(C)C(=O)N(CCCO)CCCO)ccn1C C1(CC(N2CCC(C)(C(=O)NC)C2)=O)CCN(C(=O)C=Cc2ccccc2)C1(C)C C1(C(N(C(CNC(c2nc(OCC)oc2)=O)C)C)=O)CC2C=CC1C2 Cc1nsc(C)c1C(=O)NCC1CC(C(=O)NC(C)COC(F)(F)F)CO1 c1(CC(C)C)cc(C(=O)NCC2CN(C(=O)Cc3c[nH]nc3O)C2)no1 CC1CN(C(c2ccc(F)o2)=O)CCN1C(=O)CCCn1cncn1 c1(C(=O)NC(CCC)CNC(C2(C(N)=O)CC2)=O)cccc(Cl)c1 C=CC(C)(CC)C(=O)NCC1CN(C(c2cnn(-c3ccc(Cl)cc3)c2)=O)C1 N1(C(C(C2CCC2)OC)=O)CCCC2CN(C(c3cc(N)c(Cl)c(O)n3)=O)CC12 c1(C(N2CC(NC(CCS(C)=O)=O)CC2(C)C)=O)ccc2c(c1)C(=O)NC2 S(=O)(=O)(c1ccc(-c2cccc3cccnc23)cc1Cl)N1CCCC(N)C1 C1(C(N2C3(C)CC3CC2)=O)N(C(C2CC3(CCC3O)C2)=O)CC12CCCC2 c1(CNC(C)=O)ccc(F)cc1NC1(c2nc(C(C)(C)C)no2)CC1(C)C c1(C(=O)NC2(C)CC(NC(=O)CCc3cn[nH]c3)C2)ccc(S(N)(=O)=O)c(Cl)c1 N1(C(=O)CCOCC(F)F)CCC2C(CCN2C(C2CCNC2=O)=O)C1 C1(CNC(CCN(C(C=CCCC)=O)C(C)C)=O)CCCCO1 ClC1(Cl)CC(Sc2nnnn2-c2ccccc2)C1.C1COC1 c1(C(=O)NC2CC(CNC(C(C)NC(=O)NC)=O)C2)csc(Br)c1C c1(C(=O)NC(CCOC)CNC(c2cn(CCO)nn2)=O)cccc2nn[nH]c12 CN=C(NCCC1CCSC1)N1CCC(NC(c2cccs2)=O)C1 N1(C(c2cn(CC)nn2)=O)CC(NC(C2(C(F)(F)F)CC2)=O)CC12CCCC2 c1(CNC2C(C(=O)NCc3ccccc3F)C2)cc(O)ccc1F C1(CC=C)(C(=O)NC2CC(CF)C2)CCN(C(=O)CCOCC2CC2)C1 n1(CCCOC)nnnc1C(C1(C)CCCC1)NC(C1CCOCC1)CCO C#Cc1cccc(CC(=O)Nc2cc(C)c(OC)cc2OC)c1 CN1CC=C(CNC(=O)C(C)(C)C(=O)N2CCCC2)CC1 C=C(C)CCCC(=O)N1CCC(CNC(=O)C(c2ccc(Cl)c(F)c2)O)C1 CCC(C)CC(=O)NC(C1CCN(C(c2ccc(-c3cnco3)cc2)=O)C1)(C)C C1(C(=O)NC2C(C)CCN(C(c3occ4c3CCC4)=O)C2)CC2C=CC1C21CC1 Cc1ccc(C2C(C)CN2C(=O)NC2CCOC2C)cc1 N1(C(CC(CCC)O)=O)CCCCC2(CCN(C(=O)Cc3cc(C)on3)C2)C1 c1(OC)cc(C(=O)NCCN(C(=O)Cn2cc(C(C)O)nn2)C2CC2)ncn1 CCCC(C(=O)OC)C(=O)N1CC2CCC1CN2C(=O)CCc1cnoc1 C1(NC(=O)CC2(CO)CC2)C=CCN(C(c2cnn(-c3ccncc3)c2)=O)C1 c1(C(N2CCC(NC(c3ncccn3)C)C(C)C2)=O)ccc2cccnn12 C1(CC=C)CCCCC1Nc1ncc(OCc2ccccc2)cn1 c1(CN(C)C(C2CCC(F)(F)C2O)=O)ccc2c(c1)OCO2 C(=O)(C#CC1CCCO1)NCC1(CNC(c2c(CC)[nH]cc2)=O)CC1 Cc1ccc2c(=O)c(C(=O)NC3CCC(N(C)C)CC3)c[nH]c2c1C c1(C(N(C2CCN(C(=O)CSc3n[nH]c(C)n3)C2)CCC)=O)ccc(Cl)nc1 c1(C(C(=O)N(CCNC(C2CN(C(C)C)C2)=O)C)C(=O)C2CC2)ccc(O)cc1.OC Cc1ccc(C(N2CC(C(C)NC(c3ncc(F)cc3F)=O)C2)=O)cc1[N+](=O)[O-] C#CCC(O)C(=O)N1CC2CC1C2C(=O)NC(c1cn(C)nn1)C C(=O)(CC(C)(C)CN(c1cnco1)CC1CCC1)OC Cc1ccc(SCC(C)NC(=O)C(C2(O)CCOCC2)O)cc1 C1(C(=O)NCC2(NC(=O)CN3CC(C)(C)C3)CC2)(CC)CC12CCC2 CS(=O)(=O)c1ccc(C(N2CC3=C(C2)CN(C(C2CCNC(=O)C2)=O)C3)=O)s1 N1(C(c2nc(CC)sc2N)=O)CCC(NC(=O)CCN2CCCC2)CC(C)(C)C1 C1(C)(CNC(C2OCCC(C)(C)C2)=O)CN(C(=O)Cc2ccoc2)C(C)(C)C1 C1(COc2ccccc2F)C(C)CCCN1C(=O)NCC(n1cccn1)C c1(NCC(C(CC)C)C)cc(N(C)CCOc2ccccc2)nc(C)n1 C12(C(C(C)C)NCCCSCC)CC(C(C)C)(C1)C2 C1(NC(C)=O)C2CC3CN(C(=O)CNC(=O)Nc4ccc(Br)o4)C1C3C2 CC1(CS(C)(=O)=O)CCCN(CC(c2ccncc2C(N2CCOCC2)=O)=O)C1 O=S(=O)(c1ccc(NCCC2CCOC2)cc1Cl)NCC(F)C1CCC1 C1(CC2CCC(NC(C(C)CS(C)(=O)=O)=O)C2)CCc2ccccc2O1 Cc1ccc(-n2cc(C(=O)N(C)C)nn2)cc1NC(C1CC(F)(F)CS1)=O Cc1csc(=NCC(=O)NC2(C)CC(NC(c3cc4cc(F)ccc4o3)=O)C2)[nH]1 N1(C(C2(CC)CCOC2)=O)CCCC(F)(C(=O)NOC2CCCCC2)C1 C1(C(=O)NCCCOC=C)C(O)CCN1C(=O)Nc1ccccc1C(N)=O N1(C(CCC2(C)CCCN2C(C2CCOCC2)=O)=O)CCCC2(C=CCO2)C1 c1(C(=O)NCC2N(C(C3=NNC(=O)C3)=O)CCC2)ccc2c(c1)NCC2 c1(C(=O)NCCCC2OCCN(C(C(C)(C)OC)=O)C2)cccc(S(N)(=O)=O)c1 CC1(C)CN(C(C23CC(C2)C3)=O)CC(CNC(C2CCC3C(C2)C3(F)F)=O)O1 Cc1cc(-c2nc(-c3ccccc3Br)nn2C(C)C(C)C)cc(C)c1 C1(C)(NC(CCC)=O)CCC(NC(C2(Cc3ccc(C#N)cc3)CC2)=O)CC1 N1(C(C2(C#C)CC(=O)C2)=O)Cc2occ(C(=O)NC3CC4CC(OC)C4C3)c2C1 C1(C(N(CCCNC(C2(C)CC(=C)C2)=O)Cc2ccccc2)=O)COCCN1C C(=O)(C(C)CC(C)(C)C)N1CC(NC(c2ccc(OC)c(Cl)c2)=O)C(O)C1 C1(NC(CCCC#C)=O)(CNC(c2ccc(CCO)cc2)=O)CCC(F)(F)CC1 C1(C(N2CCN(CC(=O)NCC(C)C)CC2C)=O)CC(F)(F)CCC1(C)C CC(C)(O)C(Cc1ccc(F)cc1)NC(=O)CC1C(C)(C)C1(C)C C(=O)(NNc1ccc(Cl)cc1Cl)Nc1c(C)c(N)ccc1 C(CCCC(C)(C)NC(=O)CCCN=[N+]=[N-])NC(COc1cn(C)nc1)=O c1(C(N)=O)ccc(=NCCCC(c2ccccc2)NC(=O)C2=COCCO2)[nH]c1 C12CCC(CC1)CNC2=O.N1(C(CCOCC#C)=O)CCOCC1.C(=O)(C)NC C1(CC)(CO)CCCN(C(c2sccc2CNC(c2cc(O)nc(C)n2)=O)=O)C1 CC(C(=O)NC(CNC(=O)CS(=O)(=O)C1CC1)C1CC1)C1=CCCC1 c1(NC(c2c(OC)cccc2F)=O)ccc2[nH]c(C)cc2c1 N1(C(=O)Cc2nc[nH]n2)CCN(C2CN(C(=O)COCCCCC)C2)CC1 c1(C(=O)Nc2ccc(NC(C#CC)=O)c(F)c2)cc(C#N)c2cc[nH]c2c1 Cc1cc(C(N2CCC3CC3(NC(c3ccccc3)=O)CC2)=O)n2nccc2n1 N1(C(CCC(C)SC)=O)CCN(C)CC1CNC(c1cnc(N(C)C)nc1)=O C1(NC(C=CC=CCC)=O)CCCCN(C(c2ncc(Cl)c(N)c2Cl)=O)CC1 C1(NC(C(C2CN(C(=O)Cn3ccnn3)C2)OC)=O)CCN(C)C(=O)C1 c1(CCCC)cc(C(=O)NCC2(O)CCN(C(c3ncccc3F)=O)C2)c(C)o1 C1(NC(Cc2c(C)cccc2)=O)CCCN(C(=O)COC2CCCOC2)C1C c1(C(C)NC(C2CCCN(C(c3nncn3C)C)C2)=O)nnc2n1CCCCC2 C1(CC(=O)NCC2CCC2(F)F)C2CN(C(=O)CCn3ccnn3)CC12 C1(N(C(=O)C(O)CC2CCCCC2)C)CCCN(C(C2(CO)CC2)=O)C1 c1(C(=O)OCC)cc(NC(C2C3CC(=O)CC23)=O)n(C)n1 c1(C(N2C3C(NC(C4C(C)C4)=O)C(C3)C2)=O)ccc2c(c1)CCS2(=O)=O N1(C(C(C)OCC#C)=O)CCCC2(CCCN2C(C2CC(F)(F)C2)=O)C1 c1(SC)ccc(C(=O)NCC2CCCCN2C(=O)CC2CCC(=O)NC2)cc1 C12(CC)COC(C(=O)N(CCCNC(=O)C(C3CC(C)(C)C3)OC)C3CC3)(C1)C2 C1(NC(Cn2ncc(C#N)c2)=O)CC(C(N2CC([N+](=O)[O-])C2)=O)C12CCC2 C1(NC(C(C)OCCC#C)=O)CC2CCC(C1)N2C(=O)Cc1ccccc1OC C(CCC(C(=O)Nc1cc(C)cnc1C)NC(c1cc(COC)no1)=O)OC N1(C(C(C)OCC(F)(F)F)=O)CCC(C(C)NC(C2(Cl)CC2)=O)CC1 C=CCCCC(C(=O)NC1C(C)CCC1C)NC(c1ncncc1Cl)=O N#Cc1nc[nH]c1C(N1CC2C(CNC(c3ncc[nH]c3=O)=O)C2C1)=O C12(CNC(=O)CSc3n[nH]c(O)n3)CCCCC1CN(C(=O)Cn1cnnn1)C2 C1(C(C)C)(C(=O)NC(c2c[nH]ccc2=O)C)CCN(C(c2nc[nH]n2)=O)C1 c1(C2OCCN(C(c3cccc(OC4CCC4)c3)=O)C2)cc(F)cc(F)c1 n1(CC)nc(C)c2cc(C(=O)NC3CC(C)(CNC(=O)C(O)C4CC4)C3)sc12 C1(CC#C)CCN(C(c2ccnn2CCOC)C(=O)Nc2ccc(C)cc2)CC1 c1(C(=O)NC(CN(C(C(C(=C)Cl)(C)C)=O)CC)C)cc(F)cc2c1C(=O)CC2 c1(C(=O)NC(CNC(CN(C2CCC2)C)=O)C2CCC2)ncccc1N c1(CC)cnc(O)c(C(=O)NCCCN(C(=O)CCC2CCCCC2)CC)c1 Cc1cccc(C(=O)NC2CCN(C(=O)C=Cc3nc(C)c(C)[nH]3)CC2F)c1Cl C1(C(N(CC(C(=O)NCCCn2c(C)nnc2)C)C)=O)CC(O)C(F)C1 N1(C(C(N(C)C(=O)NN2CCOCC2)C2CC2)=O)CCC(F)(C(N)=O)C1 C1(C(C(N2CCC(CNC(CSC)=O)C2)=O)C)CCC(C)(C)CC1 C(=O)(C1=C(C)OCCC1)N1CC(OC)C(NC(=O)CCCN(C)C)CC1 N12CCC(C)(C)C(C1)C2=O.c1(CC(=O)NC2C(=C)C2)scnc1-c1ccccc1 CC1CCCC(=O)CN1N1CCN(c2nsc(C(=O)O)n2)CC1 Cc1cc(C(=O)NC2CCC(NC(c3cc(N)cc(O)n3)=O)C2)c2occc2c1 N1(CCNC(c2cn(C(F)F)cn2)=O)CCN(C(C2CCS(=O)(=O)N2)=O)CC1 N1(C(c2c(C)nsc2N)=O)CCC2(CCOC2)C(CNC(C2(C)CCCO2)=O)C1 C1(C(=O)NCC(C)C(=O)NCC(c2cccnc2)O)CC2(CSC2)C1 CC1COC2(C1)CN(C(=O)C(F)CC(C)(C)NC(=O)C1=COCC1)C2 N1(C(N(CC2CCN(CC)CC2)CC)=O)CC(C)N(C(C)C)C(C)C1 C1(C(=O)NC(c2ccncc2)C)CCN(C(=O)CCc2ccc(F)cc2)C1(C)C C1(NC(c2[nH]cc(C)c2)=O)C2CC3CN(C(=O)CC4CCC(O)C4)C1C3C2 Cc1nc(C=CC(=O)NCC2COC(CNC(=O)CCN3CCCC3)C2)[nH]c1C c1(C(C)CSCC(C)N(C(C2CC(CF)C2)=O)CC)ccccc1 N1(C(C2C(C(C)C)CCC2)=O)CC2(CC(NC(c3nnc(O)cc3O)=O)CO2)C1 C12(C(N(CC(C)O)CCO)=O)CC(C)(CN1C(=O)CCn1cnnn1)C2 c1(NC(C(CCC)CNC(c2cncnc2C)=O)=O)ccc2c(c1)CCC2 C(=O)(CCCCC(F)(F)F)N1C2CC(CNC(C(C(CC)(C)C)O)=O)C1CC2 N1(C(CCC2(NC(C(C)n3cnnn3)=O)CCCC2)=O)CC(F)(F)C1C1CC1 C1(OC)CCC2(CCN(C(=O)CN(C3CCC3)C(C3CCCC(C)(C)C3)=O)C2)C1 c1(C(=O)NC2(CC=C)CN(C(c3csnc3C)=O)C2)cccc2nsnc12 Cc1nc(C(C)C)ncc1C(=O)NCC1CCCCN(C(=O)C=CC2CCC2)C1 N1C(N(C)C)=NCCSCC1.N1(CC(C)C)CCOCC1 C1(C(N2CC(C)CC(CC)C2)=O)CCN(C(c2cc(O)n(C)n2)=O)CC1(C)C N1(C(C2(COC)CCC(=O)N2)=O)CCC(NC(c2cnc(C)cn2)=O)C(F)C1 C12(NC(COc3c(OCC)cccc3)=O)CCCC1N(C(=O)C(F)=C(C)C)CC2 C(=O)(CCC(=O)NCC1CC(C)N(C(c2ccc(Br)o2)=O)C1)N(CC)CC C(C)(C(=O)NCC(C)(C)CN(C)C(c1cnc(C)nc1)=O)(C(C)C)OC C(=O)(CC(COC)NC(C1CN(C)C1)=O)N1CCC(C(CC)CC)C1 N1(C(C(c2c(C)cccc2)C)=O)CC2CC(C1)N(C(=O)C=CC(C)C)C2 CON=C(C(=O)NCC(C1CCCC1)Nc1cncc(Cl)c1Cl)c1ccco1 C(=O)(C1CCc2ccccc21)NCC1(O)CCN(C(C2(CCN(C)C)CC2)=O)C1 C(=O)(C(C(=O)N(C1CCCN(C(c2cncc(F)c2)=O)C1)CCO)OC)OCC N1(C(Cc2ccc(C)s2)=O)CC2(CCN2C(C2CCN2C(=O)OC(C)(C)C)=O)C1 CC1CN(C(c2ccc(N(C)C)cn2)=O)CC1NC(=O)C(F)(Cl)c1ccccc1 C1(NC(C2N(C(CCC)=O)CCC2)=O)CN(C(C2OCC2(C)C)=O)CC2(CCC2)C1 C(C)(CNC(=O)C(C1CCOCC1)OC)(C(C)C)NC(CCC=CCC=C)=O C1(NC(C2C(C)OCCC2)=O)CCCCN(C(c2cc(O)cnc2N)=O)C1 N1(C(c2c(C(C)C)nns2)=O)CC2CCN(C(c3ccoc3Br)=O)C2C1 C(C(C(=O)N1C2CSCC1C2)C(C)C)NC(C1(CCCC)CCC1)=O c1(C(N(C(C(=O)NCC(C)C)C)C)=O)ccc(NC=O)cc1 c1(CCC(=O)N(CC(O)CNC(=O)CN2CCCC2CO)C)c(F)cccc1F CCCS(=O)(=O)CC(=O)N1CCCCC1C(C)NC(c1ncccc1SC)=O c1(CC(=O)NC(C2(O)CCN(C(=O)Cn3ncn(C)c3=O)C2)C)cccnc1Cl N1(C(c2cnc(CC)nc2)=O)CC2(CNC(=O)CCc3nncs3)CC1CO2 N1(C(c2ccc(CC)c(C)c2)=O)CCCN(C(C2CCN(CC)C2)=O)CC1C O=c1cc(NC2CCN(c3cccc(Cl)n3)C2)nc2ccccn12 CCC(C)(COC(C)(C)C)C(=O)NC1CN(C(=O)OC2CC2c2ccnn2C)C1 N1(C(c2n(CC)ccc2)=O)CC2(CCCC2NC(C2C3CCCOC23)=O)C1 CC(C)CC(O)C(=O)NC1CC(C)(C(=O)NC(c2ncc[nH]2)CO)C1 C(C(COC)CC(=O)NCC#CCNC(=O)C(C(C)C)c1ccc(F)cc1)OC C1(C(N2CC3C(CNC(C(c4ccc(C)s4)C)=O)C3C2)=O)CN2CCN1CC2 N1(C(C(CC)NC(N)=O)=O)CCC(NC(=O)C(c2ccccc2OC)O)C(F)C1 c1(C(N2CC3C(CNCC4N(C)C(=O)CC4)(C3)C2)=O)c(F)ccc(Cl)c1F N1(CC(COc2c(OCC(F)F)ccc(OC)c2)O)C(C)(C)CCCC1(C)C C1(C(=O)NCc2occ(C)n2)C(C)OCCN1C(=O)CC1COCC(C)O1 N1(C(C(C)NC(=O)Cn2cnnn2)=O)CC2CCC(NC(=O)C3=CCC3)CC2C1 C1(C)(C(=O)NCc2cn(CC(=O)NC3CC(C)(CC)C3)nn2)CCC(=O)N1 C(=O)(C1CCc2c[nH]nc21)N1C(CN(C(CC=C=C)=O)C)COCC1 Cc1ccc(O)c(C(=O)NC2CC3CC2CC3C(N2CCC(C)(F)C2)=O)c1 N1(C(CCNC(COC)=O)=O)CC(NC(=O)COCCSCC(C)(C)C)CC1C CC(F)(C(=O)NCc1ccoc1C(=O)NCC1CCC2CC12)c1ccon1 N=c1nc(O)c(C(N2CCCCC(NC(=O)CC3COC4CC3C4)C2)=O)c[nH]1 N1(C(CCC)=O)CC2(C(=O)NCCCOC3CC3)CC1CO2 C1(C(=O)NC2(CCCNC(CC3(C)CC3(F)Cl)=O)CC2)CCCCC1O c1(CC)cccc(C(=O)NC2CCC(N(C(=O)Cn3nc(C)nc3C)C)C2)c1F CCCCCCC(O)CCC(=O)N1CCC2(CC(NC(c3c[nH]nc3C)=O)C2)C1 C1(CCC(=O)NCCN(C(C2CCC2F)=O)CC2CC2)CCCCC1 N1(c2c(CN3CCC(Oc4ccc(OC)cc4)C3)cccc2)CC(C)OC(C)C1 CCC(CC(=O)NCC1CC1NC(=O)COCCN(C)C)C(F)F C1(CC)(NC(=O)C(O)CC(C)C)CCCN(C(C2(NC(N)=O)CCCCC2)=O)C1 N1(C(c2ncc(Br)cc2F)=O)CCCC(C2CN(C(C3(CO)CCCC3)=O)C2)C1 c1(C(=O)NC2CC(CCNC(c3cn(CC=C)nc3)=O)C2)cc(F)c(F)cc1Cl CC1SCCN(C(=O)CC2(NC(c3cccnc3S)=O)CCCCC2)C1C C1(NC(CNC(=O)NC)=O)CC(NC(c2cc(CO)n(C)n2)=O)C12CCOCC2 CC#CCCCC(=O)NC(C(=O)NCC(C)(Cl)CC)C1(O)CCC1 c1(CC)cc(C(N2CC(CNC(=O)C=C(C)C3CC3)C(C)C2)=O)cc2c[nH]nc12 CCC(O)C(C)C(=O)NCC1CCCN(C(C2(C(c3ccccc3)=O)CC2)=O)C1 c1(C(=O)NC2CCC(CCNC(=O)CSC(F)F)C2)ccc(C2OCCO2)cc1 C(=O)(C1=CCCOCC1)NCC(C)(C)NC(C(=CC1CCCC1)C)=O c1(C(N2CCC(O)C(C(N3CCOC4CC34)=O)C2)=O)cc(F)c(F)c(F)c1 c1(C(N2CCN(C(CCCCOC)=O)CC2C)=O)ccn2nnnc2c1 c1(C(N2C(CNC(Cn3ncc(C)c3)=O)C(C)CC2)=O)cn(C)c2ncccc12 c1(C(=O)NCC2(CNC(c3cc(F)n[nH]3)=O)CCCC2)cnn2c1OCC2 C1(C(N2CCCC(CN(C)C(C3CCCC3(F)F)=O)C2)=O)CN2CCN1CC2 C1(NC(C2C(CCC)CCC2)=O)COCCN(C(=O)C(F)C(C)(C)O)C1 C(=O)(C(CNC(=O)C(C)Cn1cccn1)C(C)(C)C)Nc1c(CC)csc1 C1(C)(CNC(c2c(C)con2)=O)CN(CC2CCC(C(C)(C)C)CC2)CCO1 CCCC(N=c1cc(C)nc(N2CCC(C)(C)C2CC(N)=O)[nH]1)C1CCCCC1 C(=O)(CC(C)(C)CC)N1CC(O)(CN(C(c2cn(CCC)nn2)=O)C)C1 c1(C(N2CC(CCC)N(C(=O)CCN(C)CCC)CC2)=O)cc(O)cc(N)c1Cl C1(CC)C(NC(=O)CC(C)(C)CC)CCCN1C(C1CCCC12CCC2)=O C1(NC(C2ON=C(C(C)C)C2)=O)CC2CCC(C1)N2C(=O)CC1CCC(=O)N1C S(=O)(=O)(c1cccc(Cl)c1Cl)N1CC2CN(C(C(C(CC)C)N)=O)C2C1 CC1(C)CC(CNC(C2CC=CC2)=O)CN(C(C2CCC(C3CC3)CC2)=O)C1 C1(OC)CN(C(=O)C(CNC(=O)CC2CC2)C(C)(C)C)C2(CCC2)C1 C1(NC(C(CSC)O)=O)CC12CCC(NC(c1c(C)ccnc1C)=O)CC2 C(=O)(C1=CCCCC1C)NC1(CC=C)CN(C(c2ccc([N+](=O)[O-])s2)=O)C1 C1(C(=O)NCc2ccc(C(=O)NC(c3ccccc3O)C)s2)CCC(=O)CC1C C#CC1CCC(C(=O)NCC2(O)CC(NC(c3cc(Br)c[nH]3)=O)C2)CC1 C1(C)(OCC(=O)NC2C(C)C2)CN(C(=O)C(F)n2ccnc2)C1 C1(C(N(C)CC2CCN(C(CN(C)CC)=O)C2)=O)Cc2ccccc2N(C)C1=O C(=O)(C1=CCC(C)(C)CC1)N1CCC(C)C(CNC(c2cncc(N)c2)=O)C1 CC(F)(F)C(F)(F)CCS(=O)(=O)NC1CCOCC12CCCCC2 Cc1ccc(CCC(=O)N(C)CCN(C)C(C2OCCO2)=O)cn1.C1CC1 c1(OC)ccc(C(N)=O)cc1C(=O)NC1(CO)CN(C(=O)C(c2ccncc2)C)C1 C(=O)(C(CC(F)F)NC(=O)OC(C)(C)C)Nc1n[nH]c(=N)o1 n1(C(CC)(C)C)nnnc1C(c1cnc(C2CC2)o1)NCC1(C)CC1 C(=O)(C(C)(C)CC#N)NC(c1ccc(CNC(C2(CO)CC(F)(F)C2)=O)cc1)C Cc1nccn1C(C)C(=O)NCCC1CCN(C(c2cscc2C(F)F)=O)C1 C(=O)(CCCCNC(=O)C(C)(C)C1CCCN1C(C1CCN1C(C)(C)C)=O)OC c1(OC)ccc(C)c(C(N2CC3(C2)CN(C(=O)Cc2cnccc2Cl)C3)=O)c1N NC(=O)CC(O)C(=O)NC1CC(CC(=O)NC(CC2CC2)CC2CC2)C1 c12ccc(cn1)[nH]c2=O.c1(C(C)(C)N(CC(C)C)C2CC2)cc[nH]n1 C1(C(=O)NCCC#CCC)CCN(C(c2sccc2C)=O)C12CC2 C1(CC(N2CCC(C)(CNC(COCCOC)=O)C2)=O)COc2ccccc2O1 CC1(C)COC(CC(=O)NCCC2CN(C(=O)COC3COC3)C2)C1 C1(C(N)=O)CN(C(=O)C(C2CC2)NC(=O)Cn2ncnn2)CCO1 c1(C(N2CC3(N(C(CCOC)=O)CCCC3)C2)=O)oc2ccccc2c(=O)c1C Cc1[nH]nc2c1CC(C(=O)N(CCCN(C(=O)C(C1CCCCC1)F)C)C)CC2 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NCC(C)CN(C(=O)CCN(C)CCO)C Cc1ccc(C(=O)NCC2(CNC(=O)Cn3nnnc3C)CC2)c(F)c1 CCC(CNC(=O)COCCOC)(CC)NC(=O)CC1CCCC1.c1ccncc1 N1(C(C(CC)C#N)=O)CCCC(n2cc(-c3cccc(N)n3)nn2)CC1 C1(C(=O)NCC(C2CCCC2)NC(=O)NC2CC(=O)N2)CCCCC12OCCO2 c1(C(=O)NC2CCCC(NC(CC(=C=C)C)=O)C2)ccc2c(c1)CNC2=O N1(CCNC(C(N(C(COCCC)=O)C)C2CC2)=O)CC2CCC1C2 Cc1cn(C)cc1C(N1CCC(C2CCCCN2C(=O)CCN2CCCC2)C1)=O c1(C(N2CCC(CNC(C3C(=C)C3)=O)CC2)=O)sc2ccsc2c1C CC1CN(C(=O)CP(C)(C)=O)CCC1N(C(=O)CN1CC(=O)N(C)C1=O)C N1(Cc2nc(CC)oc2)CCC2(CC1)CC2C(N1CCCC(C(F)(F)F)C1)=O c1(C(=O)NC2CCC(NC(C3CCC(CC)CC3)=O)C2)cc(C(C)C)ccc1F CC(C)C(N=[N+]=[N-])C(=O)N1CCC(N(C(=O)CCc2ccsc2)CC2CC2)C1 CN(C1OCCc2sccc21)S(=O)(=O)c1cccc(OC(F)(F)F)c1 c1(C(N2CCCN(C(C(C)(F)C(F)(F)F)=O)CC2)=O)ccc(C#CC2CC2)cc1 CCCC(C(=O)N(C1CCN(C(c2ccccc2NC(N)=O)=O)C1)C)OCCF N1(C(C2(F)C(C)OCC2)=O)CCC2(C1)c1[nH]cnc1CCN2C(=O)C1=NOCC1 c1(C(=O)NCCCCNC(C2CC(CCC)OCC2)=O)cc(C)ccc1O N1(C(CS(CC)=O)=O)CC(CO)C2(C1)CN(C(c1c(C(C)C)n[nH]c1C)=O)C2 c1(C(N2CC(CCC)N(C(=O)C(F)C3CC3)CC2)=O)csc(S(N)(=O)=O)c1 C=CC(F)(F)C(=O)NCc1cc[nH]c1C(N1CCC(NC(C)=O)CC1)=O Cc1nc(CC(C)C)c(C(=O)NC2CCC(NC(=O)Cc3csc(C)n3)CC2)s1 C1(C(=O)NCc2cc(CC)no2)N(C(=O)C(N2CCOCC2)C)CC12CCCC2 C1(C2OCCO2)(OCCCC)CCOC1.C(CC(=O)NC)N(CCCC)C(C)CC C=CC(C)(CC)C(=O)N1CC(n2cc(CN3CCS(=O)(=O)CC3)nn2)C1 c1(C(=O)NC2(CC3CC3)CC2)n[nH]c2c1CN(C(C1CSC1)=O)C2 c1(C(N2CCC(N(CC(C)CC)C)C2)C(=O)NCCC)cc(F)ccn1 C1(NC(CCC(=O)N(CCC)CC)=O)C2CCC1N(C(=O)CSc1cccs1)C2 CCCCC(C(=O)NC(CC)CC(=O)OC)NC(=O)CCSCCC n1(CC)nc(C(=O)NC2CC(CNC(=O)C(F)C(C)C)CC2O)c(C)n1 c1(C(N(C)CC2(CNC(C3CCC=CCC3)=O)CC2)=O)noc2c1COCC2 CCC(COC)(C(=O)OCCCCC(=O)OC)c1ccccc1 Cc1ccc(Br)c(F)c1C(=O)NC1CC(O)C1n1cccn1 N1(CC)N=C(C(=O)NCC2(NC(c3nc(Cl)cc(N)c3Cl)=O)CC2)CCC1=O c1(C(=O)NCC2CCN(C(C=COCC)=O)CC2C)cc(F)c(C)c(N)c1F N1(C(c2c(C)cnc(F)c2)=O)CC(C)CN(C(C2(C)CNC(=O)C2)=O)CC1C C(C1SCCc2ccccc21)c1cn(C(=O)N(C(C)(C)C)CCCO)nc1 C12(NC(c3nc(Br)c[nH]3)=O)CCN(C(c3cccc(F)c3F)=O)CC1C2 c1(C(C)NC(COCCOC)=O)nc(C(=O)NCCOC(=O)C(C)(C)C)co1 C1(CNC(C2CC(=O)NC2)=O)CCN(C(=O)C=CCN(CC(F)(F)F)C)CC1F C1(C(N2CCC(OCCCNC(CC)=O)CC2)=O)CN2CCN1C(C)C2 c1(N2CCC(CC)C2)nc2c(c(=NC(C)c3cc(C)on3)[nH]1)CCCC2 Cc1cc(C(=O)NC2CC(NC(C3(CF)CCOCC3)=O)C2)ncc1Cl C1(C(=O)NCC2C(C)(C)C2(C)C)(CC)CCCN(C(=O)CCNC(C)=O)C1 S(=O)(=O)(c1c[nH]ccc1=NCC1CCCCC1N1CCCC1)N(CCC)CCO CN=C(NCC1CCOC1=O)N1CCN(Cc2cc(C)ccc2F)CC1 Cc1cc(NC(C2(C(=O)N(C)C)CC2)=O)ccc1NC(=O)Cc1ccno1 C1(CNC(CSCC)=O)CN(C(c2ccc(N)c(F)c2)=O)CCCO1 c1(C(N)=O)ccncc1NC(C1C2CC2CN1C(=O)CC12CCC(CC1)C2)=O C1(n2cc(C3N(CC)CC3)nn2)CCC(C)(C)N(C(=O)CC2CCC23CCC3)C1 N1(C(C23N(C(C4CCCC4F)=O)CCC2C3)=O)CCC(F)(F)C(F)C1 C1(NC(C2C(NC(CCCOCC=C)=O)C2)=O)CC2(CCC2)C1OC c1(OC)cnc(C(N2CC3C(N(C(=O)Cc4sc(C)cc4C)C)C3C2)=O)nc1 c1(C(=O)NCC(CC(F)(F)F)NC(=O)CC2CC(F)C2)ccc2ccccc2n1 N1(C(C2(C)CC3CC3C2)=O)CC2CCN(C(c3cncc(Cl)c3Cl)=O)C2C1 Cc1[nH]nc2c1CC(C(N1CCN(C(c3nnn(C)n3)=O)CC1C(C)C)=O)CC2 C1(CNC(CCC(=O)N(C)C)=O)COC(C)(C)CN1C(=O)C(CCS(C)=O)N(C)C C(=O)(C1CCCn2cc(C)nc21)N1CCCC2CN(C(CC(C=C)(C)O)=O)CC21 c1(CC(=O)N(C2CCN(C(=O)C(F)=CC3CC3)C2)CCC)cc(CC)co1 C(=O)(CCC1CCc2ccccc21)N1CC=C(CNC(c2c(C)noc2)=O)CC1 C1(O)(CNC(c2nnn(C)c2N)=O)CCCN(C(c2nocc2Br)=O)C1 C(C(=O)NCC(C)NC(=O)CC(F)(F)Cl)(C(C)C)c1cnc(C)s1 C1(C(N(C2CCCC(O)C2)C)=O)CC1C1CN(C(=O)C(F)(F)C2CC2)C1 C#CCC(CC#C)C(=O)NCCC1CC(OC)CN1C(=O)C(C)=C(C)C C1(C(N2CC(CNC(c3nc(C)sc3)=O)C2)=O)CCC2C1C2(F)F c1(NC(C(C)N(C(=O)C(c2cncn2C)C)CCC)=O)ccc2c[nH]nc2c1 C12CC3(CCN(CC3)C1=O)C2.c1(CNC(C=CC)=O)ccc(-c2cc[nH]n2)cc1 c1(N2CCOCC(C(=O)NCc3cccc(F)c3)C2)ncnc2sc(Br)cc12 c1(OC)ccc(CC2CC23CC3)cc1Cl.C1C(C(F)(F)F)NC(=O)N1 N1(C(c2ccc(C)nc2)=O)CCCC(O)(CN(C)C(c2cc(O)nc(Cl)c2)=O)C1 N1(C(CCc2cncc(OC)c2)=O)CC(NC(=O)CCOC2COC2)CCC1C c1(C(=O)OC)nc(=NC2CN(C(C3CC3C)=O)CC3(CCC3)C2)cc[nH]1 c1(C(=O)NCC(C)NC(c2cnn3c2CN(C)CC3)=O)cc2n(n1)CCCC2O c1(C(N2CC(O)CCC(NC(c3cnsc3)=O)C2)=O)cc2ccnc(Cl)c2[nH]1 c1(CC)cc(C)ccc1C(=O)NC1(CO)CN(C(=O)C(F)(F)C(O)C2CC2)C1 c1(C(N2CC(CN(C(=O)CCF)C)OCC2)=O)ccc2nc[nH]c2n1 c1(C(=O)NC(C)CN(C)C(C2CC3(C2)CC3F)=O)ccc2oc(O)nc2n1 c1(-c2cccc(OC)n2)c[nH]c2ncc(C(=O)N=c3ccnc(OC)[nH]3)cc12 NS(=O)(=O)c1ccccc1-c1cc(C2CC2)ccn1 CCC(CC(=O)NC1(C)CCN(C(=O)C(C)Oc2cccc(F)c2)CC1)C(F)F c1(C(N2C(CN(C(C3CC(OC)C3)=O)C)CCCC2)=O)cc2n(n1)CCNC2=O N1(C(C(C2CC2)OC)=O)CCN(C(C2(Br)CC2)=O)CC1CCO Cc1ccc(N(C)C(=O)NC(CCO)C2CC2)cc1 c1(C(c2cccc(N3C(=O)NC(CC=C)C3=O)c2)=O)c[nH]c2ccc(I)cc12 N1(C(C=CC=CCC)=O)C2CCC1C(F)C(NC(c1ccc3c(c1)OCC3)=O)C2 c1(-c2scc(C)c2)ccc2c(c1CNc1ncccc1C1CC1)OCO2 N1(C(C2N(CC)CCC2)=O)CCC2(CC1)CCN(C(=O)Cn1ccccc1=O)C2 C12(CNC(c3cc(=O)cco3)=O)CC1CN(C(=O)CC1CCCNC1)C2 c1(OCC#C)ncccc1C(=O)NCC1(CNC(c2[nH]ccc2C)=O)CCC1 c1(C(=O)NCC(CC(C)C)NC(c2cnc(C)[nH]2)=O)cc2n(c1)CCCNC2=O c1(C(N2CCC(O)(CNC(C(C)OCCC#C)=O)CC2)=O)cc(C)c(O)c(N)c1 C1(CCC(=O)NCCCCCn2cc(CC3CCNC3=O)nn2)CCCCO1 C=C(C)CN=C(NCc1ncn(C)n1)NCC1CCC12CCCO2 c1(C(=O)NC(CN(C(=O)CN2C(=O)CNC2=O)C)(C)C)ccnc(Cl)c1N C(CCN=c1[nH]cnc(Cl)c1[N+](=O)[O-])N(C(c1cc(C)c(Cl)cc1)=O)C C1(C(N2CC(C#C)(O)C2)=O)CCN(C(c2ccsc2OC)=O)CC1(C)C Cc1cc(C(=O)NCCCN(C(=O)C(c2cccc(O)c2)C)C)ncc1F c1(C(=O)NC23C(CN(C(CCOC(C)C)=O)C2)C3)ccc2c(c1)NC(=O)C(C)O2 C1(CNC(c2cnc(C(C)OC)s2)=O)CCCCCN1C(c1ccc[n+]([O-])c1)=O c1(OC)ccc(CNCCC(C2CCOCC2)C)cc1OC1CC1 C(=O)(C(C)(C(C)C)OC)N1C2(C(=O)NCC(CSC)(C)O)CC(C1)C2 c1(C(N2C(C)(C(N(CCC=C)CCOC)=O)CCC2)=O)ccc(F)c([N+](=O)[O-])c1C C(Cc1ccco1)(C(=O)N1CC(c2ccon2)C1)NC(=O)OC.C12CN(C1)C2=O O=C(CC1OCCc2ccsc21)N1CCCC1C1CCCN1C(=O)C1CC1 c1(N(C(C2CCCN(C(C)=O)C2)C(=O)NC2CCOC2)C)cccc(F)c1C c1(C(=O)NCCNS(NC(C)C)(=O)=O)ccc(O)c(OCF)c1 c1(C(=O)Nc2ccc(NC(c3c(C)c[nH]c3)=O)c(F)c2)ccc2oc(C)nc2c1 N1(C(c2cn(CCC)nc2)=O)CCOC2(CCC(Nc3ncc(F)cn3)CC2)C1 c1(C(=O)NC(CNC(CCC(C)CN(C)C)=O)CO)cccc2c1OC(C)(C)C2 CC1CCC1C(=O)NCCOCCN(C(=O)C=CC(=O)NCC1CC1)C CCCC(C(=O)NCC1CCN1C(=O)C(C)NC(=O)OC(=O)CC(C)(C)C)OC c1(CC)cc(C(=O)NC(c2ccccc2)CNC(c2cc(F)n[nH]2)=O)c(C)nn1 C1(C2(O)CCOCC2)(C(=O)NCCCC(C)NC(CCC(C)SC)=O)CC1 c1(CC)cc(C(N2CC(NC(C3CCC(CO)CC3)=O)C(O)C2)=O)n(C)n1 c1(CNC(C=CCC)=O)ccc(CCNC(=O)CN2CCCC2C)cc1 CC(C)C(O)C(C)C(=O)N(CCC(=O)Nc1cccc2c1OCO2)C(C)C N1(C(C(CNC(CSC)=O)CC2CC2)=O)CCOCC(C(C)C)C1 n1(C(C)C)ncc2c1CC(NC1CCCC13CCC3)CC2 C1(NC(C2(OC)CC2)=O)C2CN(C(C3CC(n4ccnn4)C3)=O)CC12 C(=O)(CS(=O)c1ccc(Cl)cc1)NCC1CC(C)N(C(=O)CCNC(N)=O)CC1 c1(C(N2CCC(OCCNC(c3cnn4c3OCC4)=O)C2)=O)nc(F)ccc1Cl C1(NC(C(OC)OC)=O)CC2(C1)CN(C(c1nncn1C1CC1)=O)C2 c1(CC)ccc(C)c(C(=O)NCC2CN(C(C3(OC)CC3)=O)CC2(C)C)c1 CC(C)CC(O)C(C)C(=O)NCC(C)(F)CNC(c1cc(F)cc(F)c1N)=O c1(C(N2CCN(C(=O)Cc3ccns3)C(CF)C2)=O)cn2cccc(Cl)c2n1 c1(C(=O)NC(C)(C)CNC(=O)C(C2CCCO2)C2CC2)ccc(CO)s1 CCC(C)(C)CCCC(=O)N1CCN(C(c2scc(C)c2C)=O)C(CO)C1 C1(CNC(COC2(C)CCC2)=O)CCCC(CNC(=O)CC2CC3(CC3)CO2)C1 C1(O)(CC(=O)NC2(C(=O)O)CCOCC2)CCN(C(C2(O)CC2)=O)CC1 CC(CC1CC1)CN=c1[nH]c(=NCC23CCCC2OCC3)[nH]c2cccnc12 C1(CNC(c2c(CC)scn2)=O)CN(C(c2nc(OC)ccc2Cl)=O)CCC1C c1(-c2c(OC)cc(C(=O)Nc3sncc3C#N)nc2)c(C)cc(C)cc1C C1(C)(CNC(C(=O)NCC)=O)CN(C(=O)C(C)OC2CCOC2)CC1C Cc1c(F)cc(C(=O)N(C(C)CCNC(C2CSCCS2)=O)C)c(F)c1N N1(C(C2(COC)CC2)=O)CCN(C(=O)CC2OCCC2(C)C)C(C2CC2)C1 C1(C(N(CCNC(CCC=C(C)C)=O)C)=O)CCCC(CC(F)(F)F)C1 Fc1cccc2ccnc(N3CCCN(c4ccccn4)CC3)c12 C=CCC(C(=O)N(CCCNC(=O)C1CC1)CCO)C(C)(C)C c1(-c2nn(-c3cnc(C)s3)c(C3CC(C)CO3)n2)c2ccccc2nn1C c1(N2CC(NC(CCN(C(C)=O)C)=O)C(C)C2)nc(C(C)C)cc(C)n1 C1(C(N(CCNC(CC2C(C)=NNC2=O)=O)C2CC2)=O)CC2(CCO1)CC2 C1(C(=O)NC2C(NC(=O)Cn3ccc(Br)n3)CC2)CC2(CCC2O)C1 C1(CNC(C2CCOCCN2)=O)CCCCC1(F)F N1(C(CCCCNC(COCCCOC)=O)=O)CCN(C)CC1C(C)C N1(C(C(CCC)OC)=O)CCCC(C(=O)NC(c2cnn(C)c2)CO)C1C c1(NC(C(=O)NCC2CCC(C#C)CC2)=O)ccc2cnn(CC)c2c1 c1(CC(C(=O)NC23CC(CC(F)F)(C2)C3)NC(N2CCCC2)=O)cccc(F)c1 Cc1nc(C(=O)NC(C)CCC(=O)NCC(n2ccnn2)C)c(C)o1 C1(NC(Cn2nc(C)oc2=O)=O)CCCC2CN(C(c3c(C)noc3N)=O)CC12 C12(NC(C(C)OCCOC)=O)CCC(CC1NC(=O)C=Cc1cocn1)C2 C1(NC(=O)CCC2CCCC2)CCC(O)CN(C(C2(F)CC2(Cl)Cl)=O)C1 Cc1sc(Cl)c(C(=O)NCc2cn(C3CCN(C(=O)C(C)O)C3)nn2)c1C Cc1c(NC(C2CCCN2C(c2ccccc2)=O)=O)cnn1-c1ccc(Br)cc1 C1(C(N(CC(C)SC)C)=O)CCN(C(=O)CC2(O)CCCCC2)C(C)(C)C1 C(=O)(CC(C)CCC(=O)NC1(C)CCN(C(=O)C(CO)NC(=O)C(C)C)C1)OC N(C1c2ccccc2CC1NC(=O)C1=CCCC1)C(c1c(C)cc(Cl)nc1N)=O C#CC1(C)CCCN(C(C2(C)CN(C(C3CN(C4CCC4)C3)=O)C(C)(C)C2)=O)C1 C(=O)(C1=CCCC(C)(C)C1)NCC(C)(CO)NC(CC(C)P(C)(C)=O)=O C(=O)(C1CCc2scnc21)N1CC2CCC(CNC(C(CSC)OC)=O)C2C1 c1(N2CCCC(C)(CCO)C2)nc(N2CC3CC2C3)c2c(n1)CCOC2 c1(C(N2CCC(C)(NC(=O)C(O)C3CC3)C2)=O)ccc2nc(=N)[nH]n2c1 C1(OC(C(=O)N(CC(=O)OCC)C)=O)CC(F)(F)C1(F)Cl c1(C(N2C(CN(C(C(C)=C(C)C)=O)C)CCCC2)=O)cnc2sc(C)c(C)n12 C1(CC(=O)NCCC2CN(C(C3C(CCC)C3)=O)C2)CCCC(O)C1 C1(C(N2CC(C)C(NC(c3cc(C4CC4)[nH]n3)=O)C2)=O)CCCC2CCCCC12 C(CCCCCNC(C1CCCN(C(=O)COc2cnn(C)c2)C1)=O)NC(C)=O CC1CN(C(=O)CCCCBr)CCN1Cc1ccc(O)c(Br)c1 C1(C(C)NC(=O)CCc2nncs2)CCCCN1C(=O)CCc1cnn(C)c1 c1(C(=O)NCC(C)CNC(c2cccc(N)c2Br)=O)cc2ccncc2s1 c1(OCC)ccc(F)c(C(=O)NCCC2CN(C(=O)Cc3cn[nH]c3)C2)c1F c1(NC(C2C(NC(C(C)NC(C)=O)=O)C2)=O)ccc(Cl)c(F)c1Cl c1(C(N(C2CCNCCC2C)c2ncc(C)nc2)=O)c[nH]c2ccc(F)cc12 N1(C(C2C(NC(C3(OC)CCOC3)=O)CCOC2)=O)CCN(C)C(=O)C1 C=C(C)CN=C1NCc2ccc(cc2)NCC(C)N1.C(C(F)F)OC N1(C(C(C(C)C)NC=O)=O)C(C(=O)NC2CONC2=O)C2CCCC12 C1(NC(C2N(C(N)=O)CCC2)=O)C2CN(C(c3cnn(CC4CC4)c3)=O)CC12 C1(C#N)(C(N2CCN(C(CC(C)F)=O)C(CC(F)(F)F)C2)=O)CC2(CCC2)C1 CC(C(=O)OC(C)(C)C)C(=O)NC1CCC(NC(c2cnc[nH]2)=O)CC1 c1(OC)cc(C(=O)N(C)CC#N)c(-c2cccc(COC(C)C)c2F)cn1 CN1CNC(=O)C12CN(C(=O)CCC1CCCCN(C(=O)OC(C)(C)C)C1)C2 c1(C(=O)NCCCCCN(C(CC2CCC(C)O2)=O)C(C)C)cc(Cl)n(C)n1 c1(N2CC3C(C)(C)C3C2)nc2ccsc2c(=NCC(F)F)[nH]1 N1(C(CN(C)C)=O)CC2(CC1CNC(c1c(F)ccc(F)c1Cl)=O)CC2(F)F c1(CNc2c(CC)ncc(Br)c2)cccc2c1nnn2C C(C(C)(C)CC(=O)NCc1csc(CNC(c2cc(C(C)C)nn2C)=O)n1)OC c1(C(=O)Nc2cc(F)cc(C(F)(F)F)c2Br)ccc(F)c2occc12 C1(C(=O)NC2(C)CCCN(C(c3c(C)nc(C)s3)=O)C2)CC2CC(C1)C(=O)N2 c1(OC)c(C)cc(C(N2CCN(c3ccc(F)cc3)CC2)=O)cc1Cl C12(NC(C3CCCCCC3)=O)CCC(C1)N(C(c1ccc(C(F)F)cc1F)=O)C2 C1(NC(COCc2cc(C)no2)=O)CCN(C(=O)Cc2ccnnc2O)CC1F N1(CC(=O)Nc2cccc(-c3nn[nH]n3)c2)CCc2c(O)cc(O)nc2C1 Cc1ccc(C)c(C(=O)NC2CCC2NC(=O)C(c2ccn(C)n2)C)c1 C#CCC(O)C(=O)NC1CC(CCNC(c2cnc(C(F)(F)F)nc2)=O)C1 N1(C(C(C)=CC)=O)CCCC(N(c2nnc(CCC)s2)C)C1 c1(C(N2C(C)C(NC(=O)CC(C)N(C)C)CCC2)=O)cnc2ccccc2n1 C(=O)(C1=NOC(C)(C)C1)N(C1CCCN(C(C2(S(N)(=O)=O)CC2)=O)C1)CC c1(C(=O)NCC(C2CCC2)NC(C(CC)O)=O)c[nH]c2cccc(Br)c12 c1(OCCC(=O)NCCN(C(=O)Cc2nn(C)cc2Cl)CC)ccc(F)cc1F C(=O)(C1=NOCC1)NC(CN(C)C)C(=O)NCC1(F)CCN(C)C1 N1(C(c2cnc(CC)o2)=O)CC2(CCCC2NC(=O)CC(C)P(C)(C)=O)C1 c1(C(=O)NC2C(C(N(C(C(CC)C)C)C3CC3)=O)C2(C)C)ncccc1F c1(CN2CC(C)NC(=O)C2)cnc2ccc(Cl)cn12.n12cc(cn1)C(=O)C2 c1(OC)c(F)cc(CN2CC3CCN(C(=O)CN(C)C)C3C2)cc1F c1(C(=O)NCC2(NC(C(c3c(C)n[nH]c3C)C)=O)CCC2)cc(Cl)c(F)cc1Cl CC1(C)CCN(C(c2ccc(N)cc2Cl)=O)C1CNC(=O)COC(F)F CCC(C)CCC(=O)N1CCC(N(C)C(c2cc(N)cc(O)c2)=O)CC1 C(=O)(C(CO)C(C)(C)C)NC1C2(C(=O)NCC(C3CCC3)OCC)C3CC1CC23 c1(C(N2CCOCC(NC(c3cnn[nH]3)=O)C2)=O)cc(Cl)c(Cl)c([N+](=O)[O-])c1 N1(C(C(C(C)C)n2ccnc2)=O)CC2CCN(C(c3sccc3C#N)=O)CC2C1 Nc1c(C(=O)NC2CCN(CCNC(C3C=CCC3)=O)CC2)ccc(Cl)c1F N1(C(CC2(C)CC2(F)Cl)=O)CC2(C1)SCCC2NC(C1CCCNS1(=O)=O)=O c1(C(=O)NCCC2CCCN(C(C3(CF)CCC3)=O)C2)cc2n(c1)CCSC2 Cc1ccc(CC(=O)NC2CCCCC2CNC(c2ccno2)=O)c(Cl)c1 c1(OC)ncnc(C(=O)N(C(C)CNC(C2CCN(C)C2=O)=O)C)c1F C1(NC(c2cc(CCC)on2)=O)CC(NC(c2ccns2)C)C12CCC2 c1(C(=O)NCC(CNC(C(CO)NC(N)=O)=O)F)cccc(Cl)c1O CN1CC(C(=O)NNC(=O)Nc2nccc(SCC(N3CCCC3)=O)n2)CC1=O c1(C(=O)NCCCNC(C2C(C(C)C)CCC2)=O)cn(C)nc1-c1ccccn1 C1(NC(C(CN(C)C)O)=O)C2CC1N(C(=O)CN1C(=O)CNC1=O)C2 C(=O)(C(CCS(C)(=O)=O)n1cc(C(O)C2CC2)nn1)N(CCC)CCN(C)C C1(C(C(=O)OC)(C)C)CCN(Cc2cc(OC(C)C)ncn2)CC1 CCCCC(CCCC)C(=O)N(C)Cc1noc(C2CC2)n1 C1(C(=O)NC2CCCN(C(c3sccc3C(F)F)=O)C2)CCC(C2CCC2)CC1 C(=O)(C(C)(C)C(=O)NC1(C)CN(C(C2CCCN(c3ncccn3)C2)=O)C1)NC c1(C(=O)NC2C(CNC(=O)CCCn3cncn3)C2)cncc(F)c1Cl O=C1CCCC(CC(N2CCC2CNC(c2ccc(CCO)cc2)=O)=O)C1 c1(C(=O)NC2(C(=O)NCC3CC3c3ccoc3)CC(O)C2)c[nH]c(=S)cn1 S(=O)(=O)(c1cccnc1NCC1CC1(Br)Br)NC1COCCN(C)C1 CC1N(C(=O)CC(C(F)F)NC(=O)Cc2ccn(C)n2)CCCC12CCC2 C1(CNC(=O)C2=COCC2)CC2COCC2N1C(c1coc(Br)n1)=O C12(NC(c3cc(Cl)c(Cl)[nH]3)=O)CCC(C1)N(C(C1CCCC1(F)F)=O)C2 C1(N(C(=O)C(F)(F)OCCOCCOCCOCCO)C)CCC(N)CC1.CO N1(C(c2cc(-c3ccncc3)[nH]n2)=O)CCC2CCC12CNC(C1CC(O)C1)=O c1(NC(C(c2n(C)ncc2)NC(=O)CCCN2CCC2)=O)cnc2ccnn2c1 C1(C(N(C)CC2(O)CCN(C(=O)C=C3CCCC3)CC2)=O)CCCCC12CCC2 N1(C(C(CC)O)=O)C2CCCC1CN(C(c1c(C)coc1C)=O)C2 C1(C(N2CCC(CNC(c3cccnc3S)=O)C2)=O)COc2ccccc2O1 C12(CNC(C(C)OC3COC3)=O)CC(CO1)N(C(=O)CC1(CO)CCCC1)C2 Cc1c(C(=O)N(CC(C)CNC(=O)C(C)C(C)(C)C)C)ccc(Cl)c1Cl c1(CC(=O)NCCC2CCCN2C(C2CC3(F)CC2C3)=O)ccc(Cl)cc1 N1(C(CCC(C)NC(c2c(C)ccs2)=O)=O)CCC(N=[N+]=[N-])CC1 C1(C(N2CCC(NC(C3CCC(=C)CC3)=O)C2C)=O)OCC2CCCC12 N1(C(c2c(C)ocn2)=O)CCC(N(CCO)C(C2CCCN2C2CC2)=O)CC1 N1(C(CSCCC)=O)CC2CCN(C(C3CCCS3(=O)=O)=O)CC12 Cc1ccc2occ(CC(=O)N(C(C)CCNC(=O)CN3CCC(C)C3)C)c2c1 C1(NC(C(C)=C2CC2)=O)COC2(CCN(C(c3cccc(C(C)C)c3)=O)CC2)C1 C1(CCC(=O)N(C(CC)CNC(C2CC23CCC3)=O)C)CCCC(O)C1 CCCCCC(c1nnnn1CC1CCOCC1)NCCc1cncc(Br)c1 c1(CC(=O)NCC(C)NC(c2ccc(OC(F)F)cc2)=O)cccc(F)c1O CC#CC(C)(C)NC(=O)CN(C(c1cc(CC)[nH]n1)=O)C(C)C c1(C(N2CC(N)C(c3ccccc3F)C2)=O)cc(F)cc(N=[N+]=[N-])c1 N(C1CCc2ccccc21)C(=O)Cc1c(F)c(F)cc(F)c1F Cc1nn(C)c(C)c1C(N1CCC(NC(c2n[nH]cc2C(F)(F)F)=O)C(F)C1)=O c1(C(N2CCC(CNC(C)=O)C2)C(=O)NCC2CCOC2C)cc(C)sc1C C(=O)(C(CC)CCCCC)NC1(CCNC(CSCC#C)=O)CCC1 N1(CCC)CCCC1C(=O)NCCn1ccc(C(=O)NC(C)C(C)F)c1 c1(C(=O)NC(C(=O)NC(C#C)(CC)CC)(C)CO)cccn2cncc12 N1(C(C2C(CNC(CCC3C(C)C3)=O)CC2)=O)CC2CC(CO)C(C2)C1 c1(C=O)cccc(Cl)c1.c1(C(=O)NC2C(CCOC)C2)sccc1CO C=CC(C)CC(=O)N1CC(OC)C(NC(c2ccoc2Br)=O)C1 N1(C(COCCOC)=O)CCC2(CCCCC2NC(=O)CC(C)COC)CC1 C12CCCC(CC1)CNC(=NCCN1CCCC1)N2.C(C(F)(F)F)SC(F)(F)F C1(C(=O)NC2C(=O)NOC2)CN(C(C2(c3cccc(Cl)c3)CC2)=O)CC(F)(F)C1 C1(OCC)CCN(c2nnc(-c3ccc(N(CC)CC)nc3)o2)CC1C N1(C(C2CCN(C(CC)=O)C2)=O)CC(CNC(=O)C(C)(C)CF)C(F)(F)C1 c1(C(C(C)C)=O)ccc(C(N2CCC(CN(C)C(C3CC4CC4C3)=O)C2)=O)cc1 C1(C(=O)NC2C(NC(c3c(CCC)cccc3)=O)COCC2)CN(C)CC(C)O1 c1(C(=O)NC2CN(C(C=CC=CCC)=O)CC2F)ccc2nc(OC)ccc2c1 C1(NCc2c(C)nn(C)c2Cl)CN(C(=O)CN2CCCCC2C)CCC1(F)F C(=O)(C(O)CC(C)(C)C)NC1C(C2N(C(C3(C)CCC(C)CC3)=O)CC2(F)F)C1 c1(CC)cc(C(=O)NC23CCC(CC2NC(c2cnc(O)n2C)=O)C3)ccc1Cl N1(C(C(C)C2CC2)=O)CC(C)C(C)(CNC(c2nnc(O)cc2O)=O)C1 c1(C(=O)NCC2CC(NC(c3cnc[nH]3)=O)C23CCC3)cc2c(s1)CCCC2 N1(NCCc2c(F)ccc(OC)c2)C(=O)CSC(c2cccs2)C1=O Cc1cc(C(N2CCCC(NC(=O)C(C)CO)CC2)=O)ccc1Br Cc1ccc(CNC(C2(NC(c3sccc3C#N)=O)CC(F)C2)=O)cc1 c1(C(N2CCC(O)(CC)CC2)=O)c2c(nn1C)CCN(C(C1(C)CC1C)=O)C2 Nc1cc(C(=O)NCC2CCCN(C(=O)CC3CCNC(=O)C3)C2)cnc1N N#Cc1cc2c(nc1N1CC3CC1(CNC(=O)Cc1cc[nH]n1)C3)COCC2 CCC(CC(=O)N(C1CN(C(c2c(C)ccn2C)=O)CCC1O)C)CC(F)(F)F C(c1ccccc1)=C(CC)C(=O)NCC(C1CC1)NC(C1CCCN1N=O)=O c1(C(=O)OC)cccc(CN=C(NCC(F)F)NCc2cc(C)no2)c1 c1(C(=O)NCC2C(CNC(Cc3[nH]c(=N)sc3)=O)C2)ccc(Cl)c([N+](=O)[O-])c1 c1(C(=O)NC(CCCC)CNC(C2(Cl)CC2)=O)cccc2c1OC(C)C(=O)N2 C(C)(C(C(=O)NCC1(N(C)C)CC1)C(C)C)NC(c1n[nH]c(C)c1Cl)=O C1(COC)(CO)CCN(C(=O)NC(C2CCCO2)C)C1 CC1(C)CCC=C1C(=O)NCC1CN(C(=O)CC(O)C2CCCC2)C2(CCC2)C1 n1(C(C)C)ncc2cc(C(=O)NC3CC(CNC(=O)COC(F)F)C3)cnc12 C1(CC=C)(C(=O)NC(c2ccccc2O)C)CCCN1C(c1cc(C)ncn1)=O CCC(CNC(=O)C(C)CS(C)(=O)=O)(CC)C(=O)NC1CCCC1CCO c1(C(N2CC(NC(COc3cn(C)nc3)=O)C(C)(C)C2)=O)cc2n(n1)CC(F)C2 n1(CC(=O)NCCN(C(=O)CS(=O)C(F)(F)F)C2CC2)cccc([N+](=O)[O-])c1=O c1(C(=O)O)ccc(S(=O)(=O)NC2CC(C(=O)NCC3(O)COC3)C23CCC3)s1 c1(C(=O)NCC(N2C(C(N3CC(OC(C)C)C3)=O)CC2)=O)ccc(O)cc1 c1(C(=O)NCC2(CNC(CC(CC)C)=O)CC2)c(OC)ccn2ccnc12 c1(C(N(CC(=O)NCCP(C)(C)=O)C2CCC2)=O)csc(C#N)c1 N1(C(CCSCC)=O)CCCN(C(c2ccc(N)c(F)c2Br)=O)C(C)C1 c1(C(=O)NC(C)C(CO)NC(=O)Cn2ncnn2)ccccc1C1CC1 c1(C(N2CCC(F)(C(=O)NCC#N)C2)=O)cccc2cc(CCO)ccc12 CC1=NNC(=O)C1CC(=O)NC1CN(C(c2cncn2-c2ccccc2C)=O)C1 CCC1=NOC(C(=O)NC2CN(C(c3c(C(C)C)n[nH]c3C)=O)C2)C1 c1(C(=O)NC(CCCC)CNC(C2CC2C2CCC2)=O)ccc2cc[nH]c2n1 C=CCCC(F)(F)C(=O)NCCNC(=O)Cc1ccc(C(F)F)cc1 C=CC(C)(CCOC)C(=O)NC(c1ccc([N+](=O)[O-])cc1)C1CCCC1 C(=O)(C1Cc2ccc(Cl)cc21)NCC1(NC(C2CCO2)=O)CCCCC1 C=CC(C)(C)C(=O)NC1C=CC(CNC(C2CCC(=O)N2)=O)C1 CC1CCN(C(=O)COC2COC2)CC1NC(=O)CN1CCSCC1 C=C(C)CC(C(=O)N1CCC(F)(C(=O)NC2(c3ccnn3C)CC2)C1)OC C1(OC)CC(F)CN(C(C2CCC2CNC(C2(C)C=CCC2)=O)=O)C1 C1(OC)CN(C(=O)CC2OCCCO2)CC1NC(=O)Cc1ccccc1Cl c1(C(=O)NC2CCN(C(C3CCSCC3)=O)C2)cncc2c[nH]nc12 CCC(CCC(=O)NCC1CCN(C(c2cocc2C(=O)OC)=O)C1)OC C1(c2n(CC(=C)C)nnn2)(NC2(CO)CC=CC2)CSC(C(C)C)C1 CC1CCCN(CC(C)NC(=O)NCc2ccc(C(N)=O)[nH]2)C1 CCC(C(=O)NC(=O)C(C)CCOC)C(C)O.c12cccc(c1)-c1cn-2nn1 c1(CNC(CC(COC)N)=O)cc(Br)cc2cccnc12 c1(C2(C(=O)NCCOC3CCN(C(CC=C=C)=O)C3)CCC2)ccc(Cl)c(Cl)c1 c1(C(N(CC(C)O)CC(C)O)=O)cccnc1CNC(=O)C(c1ccccc1)O C1(OC)CN(C(=O)C=Cc2cccnc2)CCC1NC(=O)C(N1CCNC1=O)C C1(C(=O)NC2N(C(C(c3cnn(C)c3)C)=O)CC2)C2CCCC1CC2 C(=O)(CCCCCCC)N1C(CC(=O)NCCC(C=C)C)CCCC1 c1(C(=O)NC2CCN(C(C)=O)C(C3CC3)C2)csc2ccc(F)cc12 C(=O)(CC(C)(C)CN(C)C)NC(C1CCN(C(Cc2n(C)ncc2Cl)=O)C1)(C)C N1(c2nnc(C)o2)CCCC2(CC(NC(=O)Cc3c(C)nn(C)c3Cl)C2)C1 CCC(CC)CC(F)C(=O)N1C2CCC(C2)C1C(=O)NCc1ncc(C)cc1C CCC(CCC(=O)NCC1CN(C(c2cn(CC(N)=O)nn2)=O)CC1O)OC Cc1nccc(C(=O)NC2CCCCC2NC(=O)C(O)CC(C)C)c1C CCCCCC(O)C(=O)N1CC(CNC(c2ccc(C(F)F)o2)=O)(OC)C1 C1(NC(c2c(C)nc[nH]2)=O)CCN(C(=O)Cc2cc(Br)cs2)CC1C c1(NC(C2C3(CN(Cc4ccc(C)cc4Cl)C3)C2)=O)cnc2ccc(Br)cc2c1 N1(C(=O)COCCF)CCC(C=CC(N2CC(n3ccnn3)C2)=O)CC1 C(=O)(C1=CCS(=O)(=O)C1)NCC12C(CN(C(CCN(C)CCO)=O)C1)C2 N(C1c2ccccc2CC1NC(=O)C(O)CF)C(c1c(C)ccc(C)n1)=O c1(CC)ccc(C(N2CCC(CN(C)C)CC2)C(=O)NC2CC2)cn1 c1(OCC(=O)NCCCCCCNC(C23CCCC2C3)=O)cccc([N+](=O)[O-])c1 c1(C(=O)NCC2C(C(=O)OC)CCC2)n[nH]c2c1CCCC2 Cc1ccc(CCNC(N2CCC3CC3C2)=O)cc1Br c1(C(=O)NC(CNC(c2n(CCCC)ncc2)=O)C)coc(=O)c2ccccc12 C(C(=O)NC(c1ccnn1C)C(N1CCC(CO)CC1)=O)(C(C)C)SCC Cc1cc(=NCCC2CN(C)C2)[nH]c(N(C)Cc2ccc(C#N)cc2)n1 c1(C(=O)NCCOc2ccc(OC(C)=O)cc2)nc(C(C)C)ncc1Cl CC(C)CCC(O)C(=O)NCCC1CC(NC(=O)C=Cc2cccc(O)c2)C1 C(c1sccc1C)=CC(N1CC(CNC(CSCC#C)=O)(OC)C1)=O C1(CNC(c2c(CC)scn2)=O)CC2CN(C(C3CCCCN3C)=O)CC12 N1(CC(=O)NCCN(C(c2ccnn2CCN(C)C)=O)CC)CCCC1=O C1(NC(C(COCC)C)=O)CN(C(c2csc(CC(F)F)n2)=O)CC1O N1(C(COCC(C)C)=O)CCN(C(=O)CC(C)C(F)F)CC1CS(C)(=O)=O c1(C(C)(C)C)noc2ncc(C(N(C[Si](C)(C)C)Cc3ccccc3)=O)cc12 N1(C(c2[nH]cc(CC)c2)=O)CCC(NC(=O)CSCc2ccccc2Cl)CC1C N1(C(CCCn2cc(C(C(C)C)O)nn2)=O)Cc2ccccc2NC(=O)C1C c1(C(C)Cc2ccccc2)nc(-c2cccc(Cl)c2)nn1C1CSC1 C1(C(N(CC(CC)CC)CC)=O)COCCN(C(c2cc(F)ccc2O)=O)C1 C(=O)(C#CC1CCCCO1)N(CC(CO)(CO)NC(C1CCCSC1)=O)C C12(CNC(CN(C(COC)=O)C)=O)CC1CN(C(=O)CC(O)C1CCCC1)C2 c1(C(C)NC(c2ccc(F)o2)=O)ccc(CNC(=O)CCc2cnc(O)[nH]2)cc1 C(=O)(C#CC1(C)CCCO1)N1CCC(C(N(C2CC3CCC2O3)C)=O)C12CCC2 N1(C(C(C)SC(F)(F)F)=O)CCOCC1CNC(=O)C=CCOC1CCOCC1 N1(C(C=CC(=O)N(C)C)=O)CCCC1C1(O)CN(C(C2CC=CCO2)=O)C1 c1(CNC(C2C(C(=O)Nc3ccc(OCCCC)cc3)C2)=O)ccc(C)c(Br)c1 c1(C(N2C(C(C)NC(=O)CC=CC(C)(C)C)CCC2)=O)cc(C#N)ccc1N CS(=O)(=O)C1CN(C(N2CCOc3cccc(Cl)c3C2)=O)C2(CCC2)C1 C1(NC(CC2(NC(C(CN(C)C)O)=O)CCC2)=O)CC2(C1)CC(C#N)C2 n1(CCOCC)nnnc1C(c1ccc(C)o1)NC(C1(C)COC1)C c1(OC)cnc(F)cc1C(=O)N(CCCCCCNC(=O)CC1CC(F)(F)C1)C C1(CNC(Cc2ncc(C)[nH]2)=O)CC(F)CN1C(=O)CCc1cccn1C C1(NC(c2c(OC)ccnc2F)=O)CN(C(=O)C(C)c2ccco2)CC(C)(C)C1 N1(C(C2CC(F)(F)C2)=O)CC2(CCC2)CC1CNC(C12CCOC1CCOC2)=O c1(CNC(C2CCC(C)S2)=O)cccc(NC(C2(c3ccno3)CCC2)=O)c1 N1(C(C(n2cc(Cl)cn2)C)=O)CCCC12CCN(C(=O)CSCC(F)F)C2 C1(O)(CC(N2C(C)(C)CC2)=O)CCN(C(C2(F)CCOCC2)=O)CC1 CC1CCC(NC(C2CCCC2(C)C)=O)CN1C(=O)CN1CCCCS1(=O)=O c1(NC(CCC2N(C(=O)OC(C)(C)C)CCC2)=O)cc(Cl)c2n[nH]cc2c1 C1(C(N2CCC(c3ccc(C)cc3)(C)C2)=O)Cc2cc(F)cc(F)c2O1 N#Cc1c(F)cc(C(=O)NC2CC(F)(F)CC2NC(C2CCC2)=O)cc1F NS(=O)(=O)c1ccc(O)c(C(N2CCOC(c3cn(C4CC4)nn3)C2)=O)c1 n1(CC(C)C(=O)N2CC(CO)(NC(c3cnn(C)c3)=O)C2)ncc2c1CCCC2 c1(CCCNS(C)(=O)=O)cn(CC(F)(F)CNC(c2cnc[nH]2)=O)nn1 Cc1ccnc(C(=O)NC2CCN(C(=O)CCC3(C)CCC(=O)N3)C2C2CC2)c1 c1(C(C(=O)NCC2N(C(c3c(CC)occ3)=O)CCC2)C)cn(C)nc1C(F)F c1(C(=O)NC(CCCNC(C2CCCC(C(=O)OC)C2)=O)C)c(F)cccc1F C=C(C)c1cccc(NC(=O)CN(C)C(c2cc(CO)on2)=O)c1 c1(C(=O)NC(CC)CN(C(C2CC23CC3)=O)CC)c(C)coc1C1CC1 c1(C(N(C)CC2(O)CN(C(C(c3cncnc3)C)=O)C2)=O)c(F)ccc(O)c1F N1(C(c2nnn(CC)c2C)=O)CC(NC(c2c(C)cnn2C)=O)CC12CCCC2 C12(NC(CCCC#CC)=O)CCCC1N(Cc1cc(Cl)ccc1C)CC2 Cc1nn2cc(C(=O)NC3CCC(CNC(c4cc[nH]c4C(C)C)=O)C3)nc2s1 CC(CC(=O)N1CC2N(C(c3cnco3)=O)CCC2(C)C1)CC(F)(F)F C(=O)(CCCC(=O)NCCC1CSCCN1C(C1CC2(CC(=O)N2)C1)=O)NCC c1(Cn2cc(COC(=N)O)nn2)ccc(C(N2CC=CCC2)=O)cc1 CC1=C(C(=O)NCCOCC(=O)NCC2OCCCC2(C)C)CCO1 C#CC1CN(C(C23CC(C(=O)OCC)(C2)C3)=O)CCN1C(=O)C=CC(C)(C)SC C=CCCCCC(=O)NC1(CCNC(c2cc(-c3ccccc3)co2)=O)CCC1 CN1CCC(C)(C(=O)NC2CC3CC(NC(C4(CCF)CCC4)=O)CC23)CC1 c1(N2C3C(NC(C4CC(C)(F)C4)=O)(CCC3)CC2)ccc([N+](=O)[O-])cc1[N+](=O)[O-] C1(NC(C2CSCC(=O)N2)=O)CN(C(=O)Cc2cccc(F)c2)CCC1CO N1(C(c2sc(C)c(Br)c2)C(=O)NC2CC2)CCC(CO)C(O)CC1 C(CNC(C1(C)CCCC1C)=O)(CC(C)C)NC(C=C(CC)CC)=O C12(NC(c3c(COC)scc3)=O)CCCCCC1N(c1nnco1)CC2 C1(NC(C2(C)CCN(c3ncc(CCC)cn3)C2)=O)CCc2ccc(O)cc2C1 c1(C(N2CCCC(NC(CC(C=C)C)=O)(CC)C2)=O)cnn2ccnc(C)c12 N1(C(C)C)CCN(CC(=O)NCCCCC(C)(C)CNC(=O)C(O)C(F)F)CC1 C(C)(C(=O)N1CC(C)(O)C1)(N(C(C1C(C(=O)OC)CC1)=O)C)C1CC1 Cn1[nH]c(=N)cc1C(=O)NCCC1CSCCN1C(=O)CC(=O)NCC1CC1 C(c1cccc(C)c1)=CC(=O)NC(CC)CC(=O)N1CCC2CC12 N1(C(C(CC(C)C)OC)=O)CCCN(C(C2CC(F)(CO)C2)=O)CC1C(C)C c1(C(=O)NCC2N(C(c3c(CC)noc3)=O)CC(O)C2)cc2sccc2n1C c1(NC(C2C(C(=O)NCC3CCCN3CC(F)(F)F)C2)=O)cccc(Br)c1 c1(OCC(=O)NC2CN(C(C3(OC)CCCC3)=O)CC2C)ccc(F)c(Cl)c1 C1(C(N(C(CNC(CCCOC(C)=O)=O)C)C)=O)CC(=C(F)F)C1 C1(C(=O)OCC)CN(C(C2(C)CCN2C(C23CC(C2)C3)=O)=O)CCN1 C1(c2ccc(C)s2)N(C(C(=O)NCC2CC2)C(C)C2CC2)CC1(C)C N1(C(C(=O)N(CCN2CC=C(C)CC2)C)=O)CCC(C)C(C(=O)NC(C)C)C1 C1(NC(C2OCCO2)=O)CCCC(NC(C2CCCC(CF)C2)=O)C1 c1(CNC(=O)OCC)ccc(C(C)NC(=O)CCN(C)CCOC)cc1 N1(C(C(C)N(C(c2cnc(OC)nc2)=O)CC)=O)CCCCC(CO)C1 C(C(CC(C)C)C(=O)N1CCC(COC)(NC(=O)C(O)C2CCC2)CC1)OC C1(C(N(C(C)CN(C(=O)Cn2cnnc2O)C)C)=O)CCOC(C(C)C)C1 N1(C(C(F)=C(C)C)=O)C2CCC(C2)C1CNC(c1nnn(C)c1N)=O CCC(C)(C)C(O)C(=O)NC(CNC(C1(CC)CCOCC1)=O)CC(F)(F)F c1(C(N2CCC(C(C(=O)NCc3c(C)nc[nH]3)C)C2)=O)cc([N+](=O)[O-])c[nH]1 c1(C(N2C(CCNC(CC(C)(F)F)=O)COCC2)=O)cccc(C(F)(F)F)c1F Cc1cncc(C=CC(=O)NCC2CCN(C(=O)C(O)CC(N)=O)C23CC3)c1 N1(C(CSC)=O)CC2CCN(C(=O)CC34CCCC3C4)CC2C1 C1(NC(C2(C)C(C)(C)C2)=O)CC(C(=O)Nc2cnn(CC3CC3)c2)CC1O N1(C(C(C)NS(CC)(=O)=O)=O)CCCC2CN(C(C3CCCCN3N=O)=O)CC12 N1(C(c2cn3nc(C)sc3n2)=O)CCN(C(=O)CN2CC(C)C2)C(C)CC1C N1(C(=O)C#CC2CCC2)CC2CCN(C(c3c[nH]nc3C3CCOC3)=O)C2C1 CC1=C(C(=O)NC2(CCNC(c3cnn(CC(F)(F)F)n3)=O)CC2)CCO1 c1(NC(C2C(NC(c3cc(CC)no3)=O)CCCC2)=O)ccccc1N=[N+]=[N-] c1(OC)ncnc(C)c1C(=O)NCC1CCC(NC(c2ccoc2Br)=O)C1 N1(Cc2cc([N+](=O)[O-])cc(F)c2)CCc2ccc(-c3cscc3[N+](=O)[O-])cc2C1 CC1OCCN(C(=O)COC2(C)CN(C(=O)CCCn3cccc3)C2)C1C Cc1cc(C#N)cc(C)c1CC(=O)NCC1(C)CCCN1C(=O)CSC(C)C Cc1cc(NC(C2(C)CCN(C)C2)=O)ccc1NC(C1CC(=O)N(O)C1)=O c1(CC)onc(C(=O)NCc2cccc(C(N3CC(C#N)C3)=O)n2)c1C C1(C(N(C)CC2(CNC(C34CC(C#N)(C3)C4)=O)CC2)=O)CC2(CCC2)CO1 c1(COC)cn(C(C)CNC(C2CN(c3ccccn3)C2)=O)nn1 c1(C(C(=O)NCCC(C)N(C(c2c(OC)csc2)=O)C)C)cccc([N+](=O)[O-])c1 C(=O)(CC1=CCOCC1)NCC1CC(NC(c2ccc(COC)o2)=O)CC1O C1(C(N(C2CCCC2)CCCNC(C(C)NC(C)=O)=O)=O)CC2(CCC2)CCO1 CC1=NOC(C(=O)NCCCNC2CCN(C(N)=O)CC2)C1C c1(C(=O)NCCC2N(C(CCCCC#C)=O)CC(OC)C2)cccc2c1OCC2 c1(C(N2CC(C)C(C)C2C)C(=O)NCCCC)cc(OC)c(OC)cc1F Cc1cc(F)ccc1NC1CC2CCC1C21CC1 CC1C(=O)N(C(N2CCC(C(C)NC(=O)OC(C)(C)C)CC2)=O)C(=O)C1C Cc1nc(Cl)[nH]c(=NC2CC23CCC(NC(C2CCCC4CC24)=O)CC3)c1Cl c1(NCC2(c3c(O)cccc3)CCOCC2)cc(=NCC2CCC=CO2)[nH]cn1 N1(CC(=O)N(CCC)C)C(=O)C2CC=CCC2C1=O.C1(=O)CO1 C(C(F)C(=O)NC(C)CCNC(=O)CCC1CCCC1)N(OCC)CC.CC C1(CNC(c2c(C)nsc2Br)=O)C(C)CCCN1C(c1cnc(S)[nH]1)=O C1(NC(=O)CCc2ccsc2)CC2CC1CN(C(c1c[nH]nc1C(F)F)=O)C2 c1(C(=O)NCC2(C(=O)Nc3cccc(C)c3)CC2)ccccc1S(N)(=O)=O C12(C(=O)NCC3C4CN(C(C5CCCCS5)=O)CC43)CC3CC(CC(C3)O1)C2 C=CCCC(C)N=c1[nH]c2c(c(=NC3CCN(CC(F)F)C3)[nH]1)CSC2 C=C(F)C1(CC(N2CCCC2C=CC(=O)NCC(F)(F)C(C)C)=O)CCC1 c1(NC(C(C2CC(NC(c3ccccc3)=O)C2)F)=O)cnc2c(c1)CCC2 Cc1cccc(Cl)c1C(=O)NC1CN(C(=O)CNC(c2ccccc2)=O)C2CC12 CC1CCC(C)(C(N2CCCC(NC(c3cnc(C(N)=O)cn3)=O)CC2)=O)CC1 N1(C(CSCC#C)=O)CCCC(C(=O)NCCC(=O)NCC)CC1 CC(O)C(C(=O)NCC1CCCN(C(c2cnn(C3COC3)c2)=O)C1)N(C)C c1(C(N2CCCC(CC(=O)NCC(C)OC)C2)=O)ccn2nccc2c1 CC1(C(=O)NCc2csc(CNC(C3CC3c3ccco3)=O)n2)CCCC(F)(F)C1 c1(C(=O)NCC(CNC(=O)C(F)(F)CC2CC2)CO)c(F)ccc2c1OCO2 C(C)(C(C(=O)N(C(C)C(N)=O)C)C(C)C)NC(CCCOC(C)=O)=O c1(Cc2nc(-c3ccc(C)o3)nn2CCCO)ccc2c(c1)OCCO2 N1(C(c2ccc(C)cn2)=O)CCN(Cc2ccc(Cl)c(C#N)c2)CC1C#N Cc1ccnn1C(C)C(=O)N1CC(OCCNC(c2cc(C(N)=O)cs2)=O)C1 c1(C(=O)NCCCN(C(c2n(CC)ncn2)=O)C)c(Br)nc2n1CCOC2 C1(CNC(c2c(CC)ccs2)=O)CC(F)CN1C(=O)CC1(C#N)CCC1 c1(OC)cc(CC(=O)NC2(CCNC(C3CCNC3=O)=O)CC2)cc(F)c1 N1(C(c2scc(C)c2C)=O)CCC2(CCCN2C(C2CC23CC(F)(F)C3)=O)C1 CC1(C)CC(N=c2[nH]c(N3C4CCC3CC(F)C4)nc3c2SCC3)CC(C)(C)O1 C(C(C)C(=O)NC1(C(=O)NC(c2noc(C)n2)CC)CSC1)SC Cc1cccc(C(=O)N(C2CCN(C(c3ncc(F)cc3F)=O)CC2C)C)c1C CC1(C)CCC(CCNC(=O)C#CCNC(c2cccc(F)c2)=O)C1 C(N=c1[nH]c(Cl)ncc1Cl)C1C2CN(C(CCc3c(C)nc(O)nc3O)=O)CC21 c1(OC)cccc(CC(O)C(=O)NCCCC2(NC(=O)Cc3ccco3)CC2)c1 C1(C(N(C2CCN(C(c3cncc(OC(F)F)c3)=O)C2)C)=O)COC(C)(C)CO1 N1(C(CNC(CNC(C(c2ccc(C)o2)C)=O)=O)=O)CCn2cnnc2C1 c1(CCC(=O)NCC2CCCN2C(=O)C=Cc2ccoc2)nc2ccccc2o1 c1(CN(c2cc(C)ncn2)C2CCNCC2O)cc(Br)ccc1I C1(CC=C)(NC(=O)COCCC)CCN(C(c2ccn(C3CCOCC3)n2)=O)C1 CCCC(CCC)CC(=O)NCC(C(C)C)NC(=O)CC1CNC(=O)O1 C1(NC(c2ccsn2)=O)CC(F)(CNC(C2CCSC2)=O)C1 N1(C(C(C)(C)OC)=O)CCOC(C(=O)NCc2ccnc(F)c2)CC1 C1(NC(=O)NCc2nnc(-c3ccccc3)o2)CC2(CCOC2)C1 c1(OCC)ccsc1C(=O)NCC(C1CCOC1)NC(c1ccn(CCF)n1)=O C12(CNC(CC(C)O)=O)CCC1CN(C(c1ccc(OC3CCCC3)cc1)=O)C2 n1(CC)cc(Cl)cc1C(=O)NCC(C)(C1CC1)Sc1ccncc1F C(c1cnn(C)c1)=CC(=O)NC(CN(C(c1n(CC)nnc1)=O)C)C C#CC1CN(C(C2CCCN2C(C2CCC(O)CN2C)=O)=O)CCO1 C1(C(N2CCCC(N(C(c3cc(C(N)=O)[nH]n3)=O)CC)C2)=O)CC2CCC(C1)O2 Cc1ccc(OCCC(=O)NC(C2CCN(C(=O)CC(C)(C)C)CC2)CO)cc1 C1(OCCCNC(C2CC(O)C2)=O)CCN(C(=O)CC2CC(F)(F)C2)CC1 c1(CCC(N2CC(NC(C3CCCCC3(F)F)=O)C2)=O)ccc(Cl)cc1F N1(C(c2nc(CC)sc2)=O)CC(NC(c2cc(C3CCOCC3)on2)=O)CC1C CC1C(NC(=O)CCCS(C)(=O)=O)C(C)CCN1C(C1CC(n2ccnn2)C1)=O N1(C(C2C(C)C2)=O)CCC2(CC1)C(NC(=O)C(c1ccc(Cl)cc1)O)CS2(=O)=O C1(CNC(C2N(CCC)CCC2)=O)CCCCC1C(=O)NCC(=O)N(C)C CC(C)C(C(=O)NCCC1CCCOC1)C(C)NC(c1cnnc(O)c1)=O CCCC(C)(C(=O)NCC1CC1)n1cc(CNc2cc(CSC)cc(N)c2)nn1 c1(C(=O)NCC2(OC)CCN(C(=O)Cc3cc[nH]n3)C2)ccc(=O)n(CCF)n1 c1(C(N2CCC(CCNC(C3=NOC(C)C3)=O)C2)=O)ccc(P(C)(C)=O)o1 N1(C(C2(C#C)CCC2)=O)CCC(C)N(C(c2ccc(N(C)C)cc2F)=O)CC1 c1(N(C(C2CC2NC2(c3ccccc3Cl)CC2)=O)C2CC2)ccccc1Br Cc1nc(O)nc(C)c1CCC(=O)N1CCC1CNC(c1cnc(N(C)C)s1)=O c1(C(C)Nc2cc(C)c(Cl)nc2)ccc(S(C)=O)cc1 C=C(C)CCC(=O)N1CCCC(CNC(c2cccc(NC3COC3)c2)=O)C1 C1(F)(C(N(CCN=[N+]=[N-])CC)=O)CN(C(c2ccc(C(C)=O)o2)=O)C1 c1(C(=O)NC2CCCC(CNC(=O)Cc3ccsn3)C2)ccn2nncc2c1 CC(C)CC(CNC(c1cc(CN(C)C)c[nH]1)=O)NC(=O)CCc1csc(=N)[nH]1 C12(CF)CC3CC1C2C3N1CCC(Nc2ccccc2)CC1 C12CCCC1NC2=O.c1(C(=O)NCC(=O)NC2(c3cc[nH]n3)CCC2)ccco1 Cc1cc(C(=O)N(C)CC2(O)CCN(C(=O)CCF)C2)cc(F)c1C c1(SC)c(C(=O)NC2CC(C)(NC(c3cccnc3S)=O)C2)cnn1C N1(c2cc(C(C)(C)C)ncn2)CCC2(CCCN(C(=O)Cn3cncn3)C2)CC1 N1(C(Cc2nnc(C)o2)=O)CCN(C(C2CC2F)=O)C(CC(F)F)C1 C(C1Cc2ccccc21)NC(c1n(CC)nnn1)c1cc(C)on1 C1(C(C)C)CCC(C(=O)N(C2CCN(C(=O)CCF)C2)Cc2ccccc2)CC1 c1(NCC(C)CC(F)(F)F)nc2ccccc2nc1N(C)CC1CC(F)(F)C1 S(=O)(=O)(c1[nH]c(=NC2CC(Cl)(Cl)C2)ccc1Br)N(C1CCCSC1)C c1(C(=O)NCCCC(C)(C)NC(C(CC)O)=O)nncc2c1CCCC2 c1(CCC)ccc(O)c(CNC(=O)CN2CC(CO)C3(CC3)C2)c1 CC1=C(C(=O)N2CCC(NC(=O)Cc3ccc(Cl)cc3)C(CO)C2)CCC1 CN1CCN(C(=O)C(=O)NC2CCC3(CC2)N=N3)C2CS(=O)(=O)CC12 N1(C(CC2(C)CN(C(=O)OC(C)(C)C)C2)=O)CCC12CN(C(=O)C(F)Cl)C2 C(=O)(C(C)Cc1cnco1)N(C)CC1CN(C(C2(C(=O)NC)CC2)=O)C1 C1(F)(CNC(C(CCC)OC)=O)CCCN(C(C2CC(C(F)(F)F)C2)=O)CC1 c1(-c2cn(CCCN(C(CC(C)C3CCCO3)=O)C)nn2)ccc(Cl)c(C#N)c1 Cc1cc(C)c(C(N2CC3CC2C3NC(C2CCCCC2C(N)=O)=O)=O)cc1N C=CC1CCCCN1C(c1cc(Br)nn1C)C(=O)NC(C)C(=O)OC Cc1cc(CNC(=O)N(C2COCC2(C)C)C)cc2c1CCC2 C1(C)(C(N2CC(OCCNC(C(OC)OC)=O)C2)=O)CCCCC1(F)F C(C)(C)(CN=c1cc(Cl)nc(C2CC2)[nH]1)NC(c1ccc2[nH]c(C)c(C)c2c1)=O CN1CCN(C(=O)C(=O)NCc2ccccc2)C(CNC(c2cnco2)=O)C1 c1(-c2sc(CNC(c3ccnc(O)c3)CCC)c(C)n2)ccccc1Cl C(=O)(CCCCCC(C)C)NC1CCN(OC(c2c(CC)n(C)cc2)=O)C(C)C1 c1(C(N2CC(F)(CC)C2)=O)cc2ccccn2n1.C12OCCC1NC2=O CC1(C)CCN(C(=O)C2=CCCCO2)C(C(=O)NCC(C)(F)F)C1 CC1=C(C(=O)NCC23CC2CN(C(c2ccoc2)=O)C3)C(C)n2ncnc2N1C C(=O)(CC(C)CC(C)(C)C)NC(C(=O)NCCC(CCC)O)(C)C C1(C(=O)NCC2CC(CNC(c3cc(OC)nn3C)=O)OC2)CN2CCN1CC2 C1(C(N2CC(N(C(C3C(C)CC3)=O)C)C(C)(C)C2)=O)CN2CCCN1CC2 N1(C(C2CC(CC)(CC)C2)=O)CCC(C2CC2)C1CNC(=O)CC1CCCCC1 C(=O)(CCCC(N)=O)NC1CC(CNC(C(c2cn(C)nc2)(F)F)=O)CC1O N1(C(C(CC)NC(C)=O)=O)CCC2(CC1)CC2CNC(=O)CCC(C)(C)OC CCC(C)C(O)C(=O)NCc1csc(CNC(=O)Cc2cocn2)n1 C(=O)(C(Cc1cccnn1)NC(=O)CCCOC(F)F)OC n1(C(C)C)cccc1C(=O)NCCC(C)N(C(=O)CC1CC1(Cl)Cl)C N1(C(c2ccccc2I)=O)CCC2(CCCC2N2CCc3nc(O)[nH]c3C2)CC1 N1(C(CCC2N(C(CCC=C)=O)CCC2)=O)CCOC(C)CC1 C1(CC(=O)NC2(C(=O)N(CC3CCC3)CC3CC3)CCCCC2)CCCC1(F)F N1(C(Cc2c(C)ncs2)=O)CC(CNC(=O)CCNc2ccccc2)C(C)C1 C(=O)(C1CCCc2ccccc21)NC1C(NC(c2cc3oc(Br)cc3[nH]2)=O)C1 C1(CNC(c2c(C)onc2)=O)CCN(C(c2cccc(CS(C)=O)c2)=O)C1(C)C CC(CC(=O)NCC1CCC(NC(=O)CCCCN2CCCCC2)C1)C(F)(F)F C1(C(=O)NCC23CC2CN(C(C2CCCCN2C)=O)C3)(OCC)CCOCC1 CC(CS(C)=O)C(=O)NC1(CC(N)=O)CCN(C(c2cnc[nH]2)=O)CC1 C(=O)(C1=NOC(CNC(C2(C#N)CCCC2)=O)C1)N(C1CCC(C)CC1)C Cc1cccc(Cl)c1C(=O)NC1CCCC1NC(c1cn(C)[nH]c1=N)=O C1(NC(C(C)Cc2cnc[nH]2)=O)(CO)CCCN(C(C2CCOC2)=O)C1 O(NC(=N)C1CN(C(N)=O)CC12CCOCC2)CC1(c2n(C)ncc2)CC1 N1(C(C2N(CC)CCC2)=O)CCN(C(C2CC2COC)=O)CC2(CC2)C1 c1(NC)ccccc1C(=O)NCC(C)NC(=O)Nc1ccnc(C(F)(F)F)c1 C#CC1(O)CC(C(N2CC(NC(=O)CC(O)c3ccccc3)C(CO)C2)=O)C1 c1(C(CNCc2n(C)nc(C(F)F)c2)O)c(Cl)cccc1Cl c1(C(=O)NC(CC)CNC(=O)CCc2ccncc2)c(C(C)C)nn(C)c1Cl c1(C(=O)NC2CCC(CNC(C(C(C)C)NS(C)(=O)=O)=O)C2)ccn(C)c(=O)c1 N=c1[nH]ccc(C(F)(F)F)c1C(N1CCNC2CC12)=O C1(CCC(=O)N(CC(C)NC(c2ccccc2OC2CC2)=O)C)CCC(=O)NC1 c1(CC(N2CCC(C3(C(F)(F)F)N=N3)CC2)=O)ccnc(C(F)(F)F)n1 N1(C(C2CC(=C)C2)C(=O)NCCCOC)CC2CCC1C2 N1(C(C(CC(C)C)O)=O)CC2CCC1C(CNC(=O)C#CC1CCCO1)C2 C(=O)(C(F)C(F)(F)F)N1CC2C(C(=O)Nc3n[nH]cc3C3CC3)C2C1 c1(C(N2CC3CC2CN3C(c2nccs2)=O)=O)ccc2nccc(Cl)c2c1 Cc1ccc(C(=O)NC2(C(=O)N(C)CCN(C)C)CC(O)C2)nc1O c1(CC)sccc1C(=O)NCC(C)N(C(=O)CCOCCOC)C C1(C(=O)OC)C2CCC1(C(=O)NC(CNC(C1CCS1(=O)=O)=O)C(C)(C)C)C2 N1(C(CC2CC(N(C)C)C2)=O)CC(F)CC1CNC(C1CC2(CCC2)C1)=O Nc1ccc(C(=O)N2C3CC2C3)c(O)c1.c1(C2C(NC(C3CC3)=O)C2)cccnc1 c1(C(=O)NC2CCC(CNC(c3cn4c(n3)SCC4)=O)C2)cn2cccnc2n1 c1(C(N2C3CCC(NC(Cc4c(C)ncs4)=O)(C3)C2)=O)cnc2snc(C)c2c1 C(=O)(C(=O)NOC)NC(CCC)CNC(=O)CSCCC(C)C C12(Cn3cc(C(C)N(C)CC4CCCC4O)nn3)CCCC1C2(F)F N1(C(C2C(C#C)C2(C)C)=O)C2CCC(C2)C1CNC(=O)CS(=O)(=O)NC1CC1 CC1CN(C(=O)Cc2ccn(C)n2)CCC1C(=O)NC1CCC(F)(F)C1 CC(C)C(F)C(=O)NCC1CCCCN1C(=O)CCOCC(F)F C=CCC(C(=O)NC1COCC1NC(c1ncoc1C)=O)C(C)C C(=O)(C(C)(C(C)C)NC(c1cc(C2CC2)no1)=O)N(C1CC(C(=O)OC)C1)C Cc1cc(C(=O)NCCCOCCCNC(C2(C#N)CCC2)=O)c(O)nn1 C1(NC(C2(CCOCC)CCCC2)=O)CN(C(C2CCCS2(=O)=O)=O)CC1C C1(C(=O)NC2(CC)CC2)CC(=O)N(CC(C)C)C1.C12(CCC1)C(=O)N(C)C2 C1(S(C)(=O)=O)(C(=O)NC2CCN(C(C3(C(C)(F)F)CC3)=O)CC2F)CC(O)C1 CCC(CC(C)C)C(=O)N(CCCNC(C1C(Cl)(Cl)C12CC2)=O)C1CC1 N1(C(C2(CCSC)CCCC2)=O)CC=C(CNC(C2CCCN2C)=O)CC1 c1(OC)c(C(=O)NC2(CNC(C3(SC)CC3)=O)CCC2)ccnc1Cl N1(C(C(CCC)C)=O)CCN(C(=O)Cn2ccc(Br)n2)CC(O)C1 C(C1OC(=O)c2ccccc21)OC(c1c(C(N)=O)coc1)=O C(CCCCC(=O)NCCCCNC(C1CCC1F)=O)N(C)C N1(C(CC#C)=O)CCC2(CCC2NC(c2ccc(C(F)(F)F)cc2)=O)CC1 C1(NC(c2n(C(C)C)ccn2)=O)CC(C2CCN(C(=O)CO)C2)C1 C1(CC)CN(C(=O)C=Cc2ccccc2C)CCC1NC(c1coc(SC)c1)=O N1(C(CCC(=C)Cl)=O)CCCC(C)(C)C1C(=O)NCC1(C)COCCO1 C1(C(=O)NC(C2CN(C(=O)CSC3CC3)C2)C)CCOC1C(F)(F)F Cn1cc(S(=O)(=O)NCC(=O)NCC2CC2CNC(C23COCC2C3)=O)cn1 N1(C(COCCCOC)=O)CCC(C)(C)C1CC(=O)NC1CCOCC1F c1(C(=O)NCC2(CNC(CC(C)n3cccn3)=O)CC2(F)F)ccc(F)cc1F c1(C(C(=O)OCC)(C)NS(=O)(=O)Cc2sccc2Cl)cc(C)ccc1F c1(OC)cn(CC(=O)NCC(C2(O)CCN(C(=O)C(C)(C)F)C2)C)c(C)cc1=O C1(NC(c2c(C)[nH]nc2C(F)F)=O)CCN(C(c2[nH]ccc2C2CC2)=O)CC1O c1(C(=O)NCC(CNC(C2(CC)CCCCC2)=O)F)nccc2ncncc12 c1(CC(=O)NC(CC)CN(C(c2nncn2C2CC2)=O)CC)cccc(F)c1F c1(C(N2C(C(N(C)Cc3cccc(C)n3)=O)C=CC2)=O)cc(C)c(O)nn1 C(CC(C(C)(C)C)NC(=O)C(N1CC2COCC2C1)=O)NC N1(C(c2c(C)coc2)=O)CC=CC(NC(=O)CNC(=O)CC2CCCC2)C1 CCC(CC(=O)N1CCCC(C)(CNC(c2nnsc2SC)=O)C1)C(C)C C(C(C(=O)NC(C)(C)CNC(=O)C=CC1CCOC1)NC(=O)OC(C)(C)C)OC N1(Cc2c(OC)cc(O)cc2)CCN(C(c2cccc(Cl)c2F)=O)C2(CC2)C1 c1(C(N(CCNC(c2c(CC(=O)OC)scc2)=O)C)=O)nn(C)cc1Br C1(NC(C2CCC(F)(F)C2)=O)CC2(C1)CC2NC(C1(O)CCOCC1)=O N#CC1(C(=O)NCC(C2CC2)NC(C2CC2C2CCC2)=O)CCOCC1 C1(CNC(C2C(CC)C2)=O)CN(C(c2ccc(C(N)=O)o2)=O)C2CCCC2O1 N1(C(c2ccc(CC)[nH]2)=O)CCOCC(C(N2CC(=O)NC(=O)C2)=O)C1 N1(C(c2c(C)ocn2)=O)CCC2C(CCN2Cc2c[nH]c3cc(Br)ccc23)C1 C1(C(=O)NC2(CC=C)CCN(C(=O)C(C(C)C)SC)CC2)CCCC(C)(C)CC1 c1(C(=O)NCCCC(CCC)NC(=O)CCC(C)OC)c2c(c[nH]c1=N)CCC2 C(CCCCC(=O)N1CCN(C(=O)C(F)n2cccn2)CC1CO)N(C)C c1(C(N(C)C)=O)ccc2ncccc2c1.C1(=O)C(C)(C)C(=O)N2CCC(C2)CN1 c1(CNC(c2ccccc2-n2cc(C3CCOC3)nn2)=O)cc(O)nc(Cl)c1 CN=c1[nH]cc(C(=O)NC(C)CCNC(=O)CCNC(=O)CC(C)C)o1 N1(C(C(CCSC)O)=O)C2CCC1CC(C(=O)NCC#CCCO)C2 c1(C(=O)NC(CC)(CNC(c2cnncc2C)=O)CC)cnn2ccnc(N)c12 C(=O)(CC1OCc2ccccc21)CC[Si](C)(C)C.N CCC(C)CC(=O)C(=O)N1CCCCC1C(C)NC(=O)CCc1ccn(C)n1 c1(C(=O)NC(C(=O)NC(C#C)(C)C2CCCC2)CC2CCCC2)cc(Cl)n(C)n1 CC1CC(CO)N1C(=O)Cn1cc(CNC(C2CCOCC2)=O)nn1 n1(CC)cc(C(=O)NC2CN(C(=O)CC3CCCOCC3)CC2C)c(C2CC2)n1 CC1CN(C(=O)CCN(C)C(C2CCC3(CCC3)C2)=O)CCC1CO c1(C(=O)NCCN2CCN(C(=O)Cc3ccccc3Cl)CC2)cncc(F)c1Cl c1(C(C)NC(=O)NCc2cc(CC)ncc2)ccc2nc(O)[nH]c2c1 CC1CC(=O)NC1C(=O)NCC12CC(NC(=O)CN3CCC(CNC)CC3)(C1)C2 C1(NC(C(c2cn(CC)nc2)=O)=O)CC(O)CN(C(=O)C(F)(F)c2cscn2)C1 C1(NC(c2c(OC)nsc2)=O)CCCC12CCN(C(=O)C(c1cccnc1)C)C2 C(=O)(C1=C(Cl)CCC1)NCCC1CC(NC(C(C(C)C)n2cnnn2)=O)C1 N1(C(C2(C)C=CCC2)=O)CC2CCC1C(CNC(c1coc(C(C)(C)C)n1)=O)C2 CC(C)(C)C(CCO)NC(C1CCC2(CC2)N1C(=O)C(Cl)Cl)=O c1(CCN2C(=O)NCCC2)ncnc2c(-c3ccccc3)nsc12 CC1CN(C(C2CC(N(C)C)C2)=O)CC1NC(=O)CCC1CCCN1C Cc1cc(Br)cc(C)c1CC(=O)N(C(c1ccc(Br)cc1)CF)C CC(C)(C)C(C(=O)N1CCCC(NC(=O)Cc2csnn2)CC1)N1CCCC1=O c1(OCCCC)ccc(COC)cc1OC(C)CCC1CCCC1 N1(C(c2ccc(C)[nH]2)=O)CC23CCCC2(C1)CN(C(c1c(Cl)csc1Cl)=O)C3 CCC(C)(C(=O)NCC(C1CCC1)NC(=O)CCCCCSC)C(N)=O CC(CNC(c1ccc(CNC(=O)OC(C)(C)C)cc1)=O)CC(F)F C12(NCC3C(CC)CCN3C(c3ccc(C(=O)NC)o3)=O)C3C4C1C1C2C3C41C c1(C(=O)NCC2CC(CNC(C3C(C)(C(C)C)C3)=O)C2)cc(Cl)cn1C CC(C)(CC(=O)N1CCC(O)C1c1ccccc1)c1ccc(F)cc1 c1(C(C(C)Nc2nnsc2Cl)OCC)ccc2ccccc2c1 C(C(C(=O)N(C)CC1(O)CCCC1)C(C)(C)C)NC(c1c(C)oc(C#N)c1)=O c1(CNC(=O)OC(C)(C)C)ccccc1CNC(c1cocc1C(N)=O)=O C(=O)(CC(CN(C)C)C(F)(F)F)N(CCCN(C(C(CSC)C)=O)C)C c1(C(=O)NC(CNC(C(COC)O)=O)(C)C(C)C)[nH]cc2c1CCS2(=O)=O c1(C(=O)NCC(C(C)C)NC(C(C)SC(C)C)=O)ccc2ccnc(Cl)c2n1 Cc1nc(C#N)c(NCC(c2nnnn2C2CC2)OC(C2CCC2)C)o1 N1(C(c2cnc(OCC)c(Cl)c2)=O)CC2CCN(C(C3(C)C=CCC3)=O)CC12 C1(C)(C(N2CCC(NC(c3c(CC)n(C)nn3)=O)(CF)C2)=O)CC(C2CC2)=NO1 CCC(C)(CCNC(c1ccn(C)n1)=O)NC(C1CCOC1C(C)C)=O c1(C(N(C2CCN(C(C(C)n3cncn3)=O)C2)CCO)=O)cc2n(c1)CCCC2 N1(C(C=C2CCC(C)C2)=O)CCC(NC(=O)CNC(N)=O)C(C)(C)C1 CC(C)C(C#N)C(=O)N1CCCN(C(C2(C)CCSCC2)=O)CC1 N1(C(C2CCCCNC2=O)=O)CCC2(CCCN(C(=O)C(F)OC(F)(F)F)C2)CC1 N1(C(C2C(C)=CCS2)=O)CCC2(CC(NC(=O)C=Cc3cncs3)CO2)C1 C1(NC(c2cc(NC(C)=O)ncc2)=O)CCN(C(=O)C(F)CC(C)C)C12CCC2 c1(CCC)cc(C(=O)NCC(c2ccccc2SC2CC2)NC(=O)CSC)ccn1 C1(NC(C(CCC)(C)CCC)=O)COC2(CCCN(C(c3cnco3)=O)C2)C1 C(=O)(C1=C(F)CN(C(CCCCCO)C(=O)NC2CCCCC2)CC1)OC C(CC(C)C)(C(=O)N1CCC(C)(CNC(C2CCC(C)(F)CC2)=O)C1)OC C=C(C)CCC(=O)NCC1(C(C)(C)C)CCN(C(=O)C(C)OOC2CCCC2)C1 C1(CCCNC(CC(C)NC(C2CC2F)=O)=O)CCCCN1C(c1ccco1)=O CCC(CCCC(=O)NCc1ccc(C)cc1F)NC(=O)Cc1cnoc1 N1(C(c2cc(CC)on2)=O)CCC(CC)CC1C(=O)NCCC(C(C)C)OC CC1CC(C)(C)CCC1(c1nnnn1C1CCCCC1)NCCl C(C(=O)NCCC1CC1)(C1=CCSC1)N(C1CCOC1)C(C)C C1(CCNC(C2C(C)C2C)=O)CCN(C(c2ccc(C3CCCO3)[nH]2)=O)CC1 c1(C(=O)NCC(C2CCCC2)NC(C(CC=C)(F)F)=O)cccc(Cl)c1[N+](=O)[O-] C1(NC(=O)CSC2CC2)CCC(Nc2ncccn2)CC1 C(=O)(CC(C)(C)NC(=O)COCCN(C)C)N1CC(CC)(OC)C1 c1(C2C(C(N3CC(F)CC(NC(=O)CC4CC4)C3)=O)C2)ccc2ccccc2c1 N1(C(C(C)NS(=O)(=O)c2cnn(C)c2)=O)C2CCC1CN(C(C1(O)CCC1)=O)C2 C(CCc1ccccc1)(C(F)(F)F)NCC(=O)NC1(CO)CCCCC1 CC1C(NC(c2cncc(CO)c2)=O)CCCN1C(c1ns[nH]c1=O)=O c1(CC(=O)NC(CNC(C(CC)C(F)(F)F)=O)C2CC2)c(C)oc2ccccc12 C1(CC=C)(NC(=O)CC2COCC2(C)C)CCN(C(=O)Cc2ccco2)C1 C(C1=C(C)CCOC1)NC(C1(CC=C)CCCN1C(c1cnc(C)n1C)=O)=O N1(C(C(C)OCCN(C)C)=O)C2CCCC1CN(C(=O)C1=NOC3COCC13)C2 C1(C(=O)NC2(CCCC)CC2)CN(C)CCN1C(=O)CCCCOC C1(NC(c2ccnnc2O)=O)CC(NC(C2C3(CC3)C23CC3)=O)C12CCOCC2 CCC(C(=O)NCC(C1CCCC1)NC(C1(C)C=CCC1)=O)NC(C)=O C(=O)CC1=CCOCC1.C1(C(N2CC(C)N(C(C)=O)CC2)=O)CC(C)(C)OC1(C)C C(C(C)(C)C(=O)NCC(O)C(=O)NC1CCC(=O)NC1)SC N1(C(C2C(C)OC(C)C2)=O)CCC2(CCC2)C(CNC(c2ccncc2F)=O)C1 c1(C(c2n(CC)nnn2)NC2CC3CC3C2)cc(C)oc1C C(=O)(CCCCCCNC(C1COCC1(C)C)=O)NC1(C(N(C)C)=O)CC1 S(=O)(=O)(c1ccc2c(c1)NC(=O)CCS2)N1CC(C)OC(C(F)(F)F)CC1 c1(C(=O)NC2C(CNC(=O)C(O)Cc3ccccn3)COC2)cncc(F)c1 N1(C(CC2CCC(=O)N2)=O)CC2CCN(C(c3scnc3Cl)=O)CC2C1 CCCC(C)(O)C(=O)NCCCOCCC(=O)NCCCCC1CCCC1 C12(CNCCCc3c(C)cccc3)CCC(CC1)NC2 C1(C)(C(N(C2CCCN(C(C(COC)OC)=O)C2)CCO)=O)CCS(=O)(=O)CC1 N1(C(C(C(C)C)(C)O)=O)CC2CC(O)C1C2NC(c1cc(C(F)(F)F)nn1C)=O c1(CC(=O)NCC(C2CCC2)NC(=O)C=Cc2cscn2)cnc2ncccn12 C12(C(=O)NCCC3OCCN(C(C4CC5CC5C4)=O)C3)CCC(CC1)CC2 CCCC(C(=O)N1CCCC1C(C)(C)NC(C1C(C)C1C)=O)OCC Cc1nc(C)c(C(=O)N(C)CC2(O)CN(C(=O)CCC3CCCN3C)C2)o1 N1(CC(C)S(C)=O)C(=O)CCN(CC23CCC(CC2)OC3)C1=O C1(CNC(=O)Nc2sc(Br)c(C)c2C)CC2(C1)C(F)(F)C21CC1 C1(NC(=O)CCF)COC2(CCN(C(=O)CCc3cnc4ncccn34)CC2)C1 C1(CC)C(C)CCN1C(c1cnc(CONC(c2cc(C(C)C)on2)=O)nc1)=O C(=O)(CCC(=O)NC1CCOCC1C(=O)NC(c1ncco1)C)NCC CON1CC(C(=O)NC(C(=O)N(C)CCOCCO)C(C)C)CC1=O C1(CNC(=O)Cc2cccc(Br)c2)CC2(CCC2)CN1C(c1cc[nH]c1)=O Cc1ccc([N+](=O)[O-])cc1C(N1CC(C)(C(=O)NCCCn2ccnc2)C1)=O S(=O)(=O)(c1cccc(-c2cc3c(cc2O)OCO3)c1)N1CCC(C=C)CC1 c1(C(C)C)cc(C(N2CC(NC(=O)CC(C)F)CC(C)C2)=O)cc(O)n1 C1(CC(=O)NCC(C)CNC(c2cn(C)nn2)=O)CCC(C)(C)C1 Cc1cc(C(=O)NCCN(C(=O)C(c2ccc(Cl)cc2)N(C)C)C)c(C)nc1C C1(C(N(CC(CC)NC(c2c(C)noc2N)=O)C)=O)CCc2cnn(C)c2C1 C(=O)(C(C(C)(C)C)OC)OCC1(COC)CCN(C(c2cc(=O)n(C)cn2)=O)C1 N1(C(C(CCC#C)NC(=O)C(C#N)CC)=O)CC2CC(F)CC2C1 CC(C)C(CN(C)C)C(=O)N1CCCC(CNC(c2ccnnc2O)=O)CC1 CN=C(NCc1ccc2cc(C)[nH]c2c1)N1CCC(CC)C1 Cc1cc2[nH]c(C(N3CCC(O)(CCNC(c4cncn4C)=O)CC3)=O)cc2s1 C(CCC(C)(C)NC(=O)CCC1CCC(C)O1)NC(C1(CC=C)COC1)=O N1(CC(=O)N(C)CC2CCN(C(c3cnn(C)n3)=O)CC2)CCP(C)(=O)CC1 C1(NC(C=C(C)C(F)F)=O)CCCC(NC(c2cc(-c3ccccc3)no2)=O)C1 c1(N2CCC(C)(C(N)=O)C2)ncc(C(=O)O)n2cncc12 C1(C(N(CC(=O)OCC)C)=O)(NC(C2CN(C)C2)=O)CCCC1C C(=O)(C1c2c[nH]nc2CCC1C)NC(CNC(C1(C)CC(=C)C1)=O)CC C1(C(=O)NC2C(C(=O)NC(C(=O)OCCC)C)CC2)CC2(CCC2)CO1 CC(C)CCC(=O)NC1(C(=O)NCC2CCCCC2NCC23CCC2CC3)CC1 C(=O)(C(C(=O)N1CCC(N(C(=O)CCc2ccccn2)C)C1)C1CC1)OCC N1(C(c2c(C)nc[nH]2)=O)CC2C(NCc3ccc(-c4ccccc4F)o3)C2C1 c1(C(=O)Nc2ccc(-c3cncc(OC)c3)nc2)ccc2[nH]c(=O)ccc2c1 c1(CCC)ccc(NC(C2C=CCN2C(=O)C(O)C2CC2)=O)cc1 c1(C(N(CCOCCCN(C(CC(CC)C)=O)C)C)=O)cnn2c1OCC2 C1(CNC(C2C(C)C(=O)C2)=O)CCC(=O)N1C C1(NC(C(C)=C(CC)C)=O)CC(NC(=O)Cn2nc(C)c(Cl)c2C)C12CCC2 CC(C)(C)C(CNC(C1(C(N)=O)CCC1)=O)C(=O)N1CC(OCC(F)F)C1 C1(CC(=O)N(C(C(=O)OC)C)C2CC2)CN(C(=O)C(F)CC2CCOC2)CCC1C O=C1CS(=O)(=O)CC(C(=O)NC2CCN(C(c3ccc(O)cn3)=O)CC2CO)N1 C1(CCCNC(Cc2n(C(C)C)ncc2)=O)CCN(C(=O)CS(N)(=O)=O)CC1 c1(CC(=O)NCC2CCN(CC(=O)NCC)C2)c(F)cccc1F c1(OC(C2(N)CC(OC)C2)=O)ccc(CN(C)C)cc1 c1(C(N2CCC(NC(C3=CC(C)(CC)C3)=O)C(F)C2)=O)ccc2n[nH]cc2c1Cl C(N=c1[nH]c2c(c(=NCCCOC3CC3)[nH]1)CSC2)c1cc(C)c(F)cc1Br c1(CSc2c(-c3onc(N4CCCC(C)C4)n3)cccc2)n[nH]c2c1COCC2 Cc1c(Cl)ccnc1C(=O)NC1(CF)CCN(C(=O)Cc2cc[nH]c(=N)c2)C1 c1(C(=O)NCCCNC(C2(C)ON=C(C)C2)=O)ccc2c(c1)CCC(C)N2 C1(CNC(C(=O)NC2(C)CCN(C(=O)C(F)(F)F)C2)=O)COc2ccccc2C1 C1(C(=O)NCC(COC)C)CCN(C(c2cnc(OC)cn2)=O)C(C)(C)C1 c1(C(=O)Nc2ncc(-c3ccc(N4CCOCC4)nc3)s2)cc(Cl)cnc1O C1(NC(C2C(C(C)O)C2)=O)CCCCC1CNC(C1CCC(F)C1)=O c1(C2C(C(=O)NCCN(C(=O)C(C)C)CC)C2)ccccc1C(=O)OC(C)(C)C C1(C(N(CCNC(C2(C)CCN(C)C2=O)=O)C2CC2)=O)CCC(F)(F)CC1(C)C C1(C)(COC)CC(NC(c2cnc(Cl)c(N)c2)=O)CN1C(c1n[nH]cc1C)=O C(c1ccc(F)c(F)c1)=CC(N1CCCN(C(CCCCC#N)=O)CC1)=O C#CCC(C)(CC)C(=O)NCCOC1CCN(C(C2(C)CCCCO2)=O)C1 N1(C(=O)CCC2CCCO2)CCN(C(c2cn(CCC3CC3)nn2)=O)C2(CC2)C1 C(=O)(C(C)(C)Cc1ccccc1Br)NC(COC(C)C)C CC12C3C4C1C1C2C3C41C(=O)NCC(CO)NC(=O)C#CC1CCCO1 N1(C(C(C(C)C)O)=O)CC(NC(C2CC(OC(F)(F)F)C2)=O)C2CCCCC12 c1(C(N(CC(CNC(C(CC#C)C2CC2)=O)(C)C)C)=O)ncnc(C)c1OC Cc1csc(C(=O)NCCCN2CCC(NC(C3CC(CF)C3)=O)C2)c1C C1(CC)CN(C(=O)CCn2ccnc2)CCC1NC(c1cc(O)ncn1)=O Cc1c(F)ccc(Cl)c1C(=O)NCC(C)(C)NC(=O)CC(C)C1CCCO1 CC(C)(C)C1=NOC(C(=O)NC2CCCCC2CNC(C2CC3C=CC2C3)=O)C1 Cc1c(C(N2CCCC(N(C(=O)CC(C)(C)N(C)C)C)CC2)=O)c[nH]c1C#N S1(=O)(=O)c2ccc(C#N)c(c2)NCCN2CCC(CC2)N1.C(CCF)[SH](C)N Cc1cc(C(=O)NC2CN(C(C34CCCCN3CCC4)=O)CC2C)c(C)c(C)c1 c1(CNC(C2C(NC(c3ccc(O)nc3)=O)CCC2)=O)c(F)ccc(O)c1F c1(CC(=O)NC23CC2CN(C(c2scnc2Cl)=O)C3)ccc(F)cc1F c1(C(N2C(C)COCCC2)=O)nc2ccccc2cc1Cl N1(C(=O)C)CCc2ccccc2C1.C1(N2CC3CCC2C3)CS(=O)(=O)CC1O c1(OC)cc(Cl)ccc1C(=O)NC1CCCC(NC(C2(C)C=CCC2)=O)C1 C(=O)(C1OCCn2ccnc21)NCc1scc(CNC(=O)CC(C2CC2)C2CC2)n1 Cc1ccc(C)c(C(=O)NCC2CCN(C(c3cccc(CS(C)=O)c3)=O)C2)n1 C(=O)(CCCCCCC)N1C(CC(N2CC(CC#C)OCC2)=O)CC(C)(C)C1 Cc1[nH]nc2c(C(N3CCCC(C)(C)C3CNC(=O)CO)=O)cccc12 N1(C(CN(CCC)C)=O)CC2C(C(=O)NC(C)CCC3CC3)C2C1 CC1OCCC1(F)NC(=O)NC(C1CN(Cc2noc(-c3ccccn3)n2)C1)C CN=c1[nH]cc(C(N2CC(NC(c3cc(C(F)F)nn3C)=O)C3CC23)=O)s1 C1(CC(=O)NCc2c(C)csc2)C2CCC(C2)N1C(C1CN(C)C1)=O Cc1nc2c(o1)CCN(C(C1CSCN1C(C1(C)CCCC1O)=O)=O)C2 N1(C(c2nn(C)c(Cl)c2)=O)C2CCC1CC(NC(c1cncn1C1CC1)=O)C2 C(C(F)(C(=O)NC1CCn2ccnc2C1)C(C)C)NC(C(CC(C)C)=O)=O C1(C2(O)CCN(C(C3CCC(C)(C)C3)=O)CC2)(NC(c2c(C)ccnc2)=O)CC1 N1(C(c2cnc(C(C)O)s2)=O)CCCC2C1CCCN2C(C1CCC(C)CC1)=O C1(C2CCN(C(c3ccc(N4CCC4)cc3)=O)C2)(NC(C2CC3CC3C2)=O)CC1 C1(CCC)(NC(c2coc(CC)n2)=O)CCCN(C(=O)C(C)S(N)(=O)=O)C1 c1(C(N2CC(NC(Cc3c(OCC)cccc3)=O)C(O)C2)=O)cc(C)ccc1I C1(C#N)(C(=O)NC(C(C)NC(C2C(C)OCC2)=O)CO)CC=CC1 c1(CNc2n(CC(=O)O)nc(C(F)(F)F)c2)ccc2nc(O)[nH]c2c1 CCC(C)CCC(=O)N(CC(C)NC(=O)Cc1csc(NS(C)(=O)=O)n1)CC c1(CC)ccc(-c2nc(CC(=O)NCCNC3CCC3)cs2)cc1 c1(C(=O)NC2(CC(=O)Nc3ccc(I)c(O)c3)CCC2)cc(Cl)cc(Cl)n1 C1(C(N(CC(C)NC(=O)C(N)=O)CC)=O)CCN(c2cccc(OC)c2)C1=O N1(C(CC2C(NC(c3c(CC)c[nH]c3)=O)CC2O)=O)CCC(O)(CC(C)C)C1 C1(C(N(C2CCCN(C(C3(C)CCCC3)=O)C2)C)=O)CCN(S(=O)(=O)N(C)C)C1 N1(C(C(CC)CC)=O)CC=C(CC(=O)N(c2cccc(F)c2)C)CC1 c1(CN2C(C(N(C3CCC3)CC)=O)CC(F)C2)c[nH]c2cccc(F)c12 C=CCC(C(=O)Nc1ccc(-n2cc(C(C3CCC3)C3CC3)nn2)cc1)OC Cc1cccc(OCC(=O)NCC2CCCC2NC(c2cn(C)nn2)=O)c1F C1(NC(C(CCCC)O)=O)CCCCN(C(c2cncc(C3CC3)c2)=O)CC1 c1(NC(C2CC(O)(CNC(C(C=C)OC)=O)C2)=O)cnc2ncnn2c1 c1(C(=O)NCC23C(CN(C(C4(C)CC(F)C4)=O)C2)C3)cnc2nccnc2c1 c1(C(N2CC3CN(Cc4ccc(F)cn4)CC3C2)=O)c[nH]c2nccc-2c1 c1(C(N2CC3N(c4c(OC)cnc(SC)n4)C3C2)=O)cc2ccc(Cl)cc2nn1 c1(C(N2CCC(CC3CC3)C2)C(=O)NCC(F)F)cn2c(Br)cnc2s1 c1(CC)ncc(C(=O)NC2CC(NC(c3cc(C)ns3)=O)C23CCC3)c(O)n1 c1(C(c2n(CCC)nnn2)NC2CCC(C(N)=O)CC2)ccc2ncccc2c1 c1(-c2nc(-c3cccc(CO)c3)nn2C2CC2)cc(Cl)nnc1O c1(OC)cc(C)ccc1NC(c1ccc(CO)o1)c1nnnn1C1COC1 n1(C(C)C)cc2ncc(C(=O)NC3CCN(C(=O)CCC4CC4)CC3O)cc2n1 C=CC1(C(=O)N(C2CCCC2C#N)C)CCN(C(=O)CN2CCSCC2)CC1 c1(CC)nonc1C(=O)NCCCCC1CN(C(=O)C(C2CC2)C2CC2)C1 CCN=c1[nH]c(C)c(C(=O)NCCNC(C2(C)CCC(N(C)C)C2)=O)s1 C1(CNC(C(c2cccnc2)C)=O)CC2(CC(NC(=O)CCc3cncs3)C2)C1 C1(C(=O)NC2C(CNC(=O)CCCn3cncn3)C2)CCCC12CCC2 C1(C2CC2)(CNC(c2c(CCC)nco2)=O)CCN(C(=O)CCCC#N)C1 C1(NC(c2cnn(C(C)C)c2F)=O)(CO)CCCN(C(=O)CC2CC3(CC3)C2)C1 C(CC(C(C)(C)C)NC(c1cn(C)nn1)=O)N(C)C(C1CCCNC1=O)=O CS(=O)(=O)C1CC(C(=O)NCC2CC(NC(=O)Cc3cc[nH]n3)C2)C1 N1(C(CCC(=C)C)=O)CCCC2(CCN(C(C)C(=O)NC(C)CC)C2)C1 c1(CN(C(c2sncc2C)C(=O)NC(CC)(C)C)C)cc(C#N)cs1 C=CCC(C)(CC=C)NC(C1CCC(C2CC2)N1C(c1ccn(C)n1)=O)=O c1(CC(=O)NC2(CO)CCN(C(=O)CC34CCCC3C4)C2)ncc(Cl)cc1F N1(C(C(CC)(C)C)=O)CCC(C2CCCN(C(C3CC(=O)NC(=O)N3)=O)C2)C1 C(c1ccc(C)c(C)c1)=CC(N1CC(NC(CC2(COC)CC2)=O)C(OC)C1)=O Cc1c(Br)ccnc1C(=O)NC1CC(CO)N(C(=O)C(F)CC2CC2)C1 c1(C(N(CC(C)NC(C2(COC)CCCO2)=O)C)=O)ccc(C2(C)CC2)cc1 N1(C(CC=C)=O)CC2CCN(C(c3cc(N4CCCC4)ccn3)=O)C2C1 N1(C(c2c(-c3cccc(NC(COC)=O)c3)c[nH]n2)=O)CCN(C)C(=O)C1 c1(C(N(CCCOCCNC(=O)C=Cc2ccsc2)C)=O)ncncc1Cl Cc1cccc(C)c1-n1nc(CCO)nc1-c1cnc(-c2ccccc2)o1 c1(OC)cc(F)ccc1C(=O)NC1CCC(N(C(=O)CSCCN(C)C)C)C1 N1(C(CCc2ccc(CC)cc2)=O)CCCCC(CNC(c2ncccn2)=O)C1 CC(CCC1CCC1)NC(=O)CC=CCNC(=O)C=CCO C1(CNC(CCCCCSC)=O)COC(C)(C)CN1C(C1CCC(C)(C)O1)=O Cc1ccsc1CCCC(=O)N(CC(C)NC(=O)CCCOC(C)C)C Cc1ccc(C(C)CC(N2CCC(C)(NC(C3COC(C)(C)O3)=O)C2)=O)cc1 CC1CCCC(CC(=O)NC(C2CCN(C(=O)CC3CCCC(=O)N3)C2)C)C1 c1(CC(=O)NC(C2CCCC2)CNC(CN(CCC)C)=O)c(C)cc(C)nc1O C1(C(=O)NC(C=C)CO)CCN(C(c2c[nH]nc2-c2cnn(CC)c2)=O)C1 c1(C(=O)NCC(CC)NC(C2CCC(OC)C2)=O)sc(S(N)(=O)=O)cc1C C1(N(C)C)CCC(C(=O)NCCCCNC(=O)CO)C1 c1(OC)ccc(F)cc1C(N1CC(NC(c2cc(C)ccc2Cl)=O)CC1C)=O CC#CC1CCN(C(C2CCN(C(=O)C3=CCC(C)CC3)C2CC)=O)CC1 Cc1ccccc1C(C)C(=O)NCCC1CCCN1C(C1CCC1C(C)(C)C)=O c1cncc(NC(=O)C(C(C)C)N)n1.C(CN(CCNC(C)=O)C(C)=O)OC Cc1cccc(Br)c1C(C(=O)N(C(C)C(F)F)C)NC(C1COCCN1C)=O CCCCC(CC)C(=O)NC(C(=O)NCC1CC2CCC(C1)C2)C(C)(C)C CCC(O)C(F)(F)C(=O)NC12CCCC1N(C(C1CCCN1C(C)C)=O)CC2 C12(C(N3CC(CNC(c4cc(C)sc4)=O)C4(C3)CC4)=O)CCC(F)(CC1)CC2 Cc1nnc(O)c(C(N2CC3CC3(CNC(C3CN(CC(C)C)C3)=O)C2)=O)c1C c1(C(=O)NCC2CC(NC(C(CC)(F)F)=O)C2)cc(C2(C)CC2)ccc1F N1(C(CC2C(C)C2)=O)CCc2[nH]nc(CNC(c3cccc(C(F)F)c3)=O)c2C1 C=CCCC(C(=O)NCc1cc(C(N)=O)no1)NC(=O)C(F)C1CCCC1 N1(C(c2c(OC)nsc2)=O)CC(N(C(=O)Cc2ccnn2C)C)C(C)(C)C1 C(=O)(C(O)C1CC1)NCCCN(C(=O)CCc1cc[nH]n1)C c1(N(S(=O)(=O)CC)C)cc(Br)ccc1S(=O)(=O)NCC(C)OCC(O)C1CC1 c1(C(N2CCN(C)C(CNC(C3COCCO3)=O)C2)=O)cc(Cl)c(N)c(Cl)c1 c1(C(N2C(C(=O)NCc3c(C)noc3C)C(O)CC2)=O)ccc2ccccc2n1 c1(C(=O)NCC(C(C)C)NC(=O)Cn2cc(Cl)cn2)ccc2ncnc(O)c2c1 C(C(CNC(=O)C(=O)Nc1ccccc1)C(F)(F)F)NC(C(C)O)=O N1(C(Cc2cccc(CC)c2)=O)CC(F)(F)CC1(C)CNC(c1cc(C)co1)=O C#Cc1cccc(C(N2CCCC(O)(CNC(C3(CC)CCOC3)=O)C2)=O)c1F C1(CNC(CS(CC)=O)=O)CCN(C(c2cc(C(=O)OC)n(C)c2)=O)C1(C)C CC(C)CC(C)(CNC(C1(C)CC2CC2C1)=O)NC(C1CCC2(CC1)CC2)=O CCC(C)(CC)C(=O)NCc1cccnc1CNC(=O)Cc1ccccc1C c1(C(=O)NCC(C(=O)N(CC=C)CCO)O)ccc(F)c(F)c1 C1(COC)CCCCN1C(=O)CC1CCN(C(=O)CN(C)C2CC2)CC1 C1(NC(c2c(SCC)cccc2)=O)CCN(C(c2[nH]c(O)nc2C)=O)CC(O)C1 C1(C(=O)NC2C(CNC(C3CC4(C3)CC(O)C4)=O)C2)CC(c2ccncc2)=NO1 Cn1c(C(=O)NCC(C(C)(C)C)NC(C2(CO)CCCC2)=O)cnc1O CC1(C)CC(C)(CNC(c2cnsc2)=O)CN1C(=O)CC1CCCO1 C1(N(C(C(C)CF)=O)C)CCCCC1N(C)C(c1ccc(-c2ccco2)nc1)=O N1(C(C(C)OC(C)(C)C)=O)CC2(C1)CN(C(C1CC1c1cnc[nH]1)=O)CC2CO N1(C(C2CC(NC(c3cc(OC)cc(Br)c3)=O)C2)=O)CCc2ncccc2C1 C(=O)(C(F)(F)CC(C)C)N(CCC)CCNC(c1nccc(Cl)c1Cl)=O N1(C(c2cscc2C)C(=O)NC(CC)(C)C)CCCC(CNC(C)=O)C1 c1(C(N2C(C(N3C(C(=O)OC)CC3)=O)C=CC2)=O)cccc(=O)n1C CC(C)C(C(=O)NCCC[Si](C)(C)C)C(C)NC(C1CC2(CC(=O)C2)C1)=O c1(OCC=C)ccc(Cl)nc1C(=O)N(C)CC1CCN(C(=O)CC#N)C1 C(=O)(C(O)C1=CCCCC1)ON1CC(n2cc(C3CC(OC)C3)nn2)C1 C1(C(N2C(C(N)=O)CNC(=O)C2)=O)CCCN(C(c2cc3occc3[nH]2)=O)CC1 C(=O)(NN1CCCC1C(=O)NC(N1CC(CC2CC2)C1)=O)c1c(SC)nccc1 Cc1cc(C(=O)NCC2(NC(=O)C(c3cccc(F)c3)F)CCOCC2)[nH]c1C c1(N(C)C)ccc(C(N2CC=CC(NC(=O)Cc3csc(NC=O)n3)C2)=O)cn1 c1(C(=O)NC(C(C)NC(c2cnc(C(C)C)[nH]2)=O)C)cc2c(cc1Cl)NC(=O)C2 O=S(=O)(c1c[nH]ccc1=NCc1ccsc1Cl)NC1(c2ccc(F)cc2F)CC1 N1(C(CN(CC#C)C(c2ccc(CO)cc2)=O)=O)CC2COC(=O)C2C1 N1(C(CCOCC)=O)CC(NC(=O)C2=CCCC(C)(C)C2)CC2(CCOCC2)C1 c1(C(=O)NCC2(C)CCCN2C(C2CC2F)=O)cc([N+](=O)[O-])ccc1SCCO C1(NC(CC2(C)CC2)=O)CC2(CCN(C(c3n[nH]c4c3CCOC4)=O)CC2)C1 C(=O)(CCCC(F)(F)F)NC1(CO)CN(C(c2c(C)[nH]nc2C(F)(F)F)=O)C1 C(=O)(CCC(C)(C)N(C)C)NC(CNC(c1c(CC=C)cccc1)=O)CC C1(n2cc(CC)nn2)CCC(CC2CCN(C(=O)Cn3cc(Br)c(C)n3)C2)CC1 N1(CCNC(c2c(C)cc(Br)o2)=O)CC(C)(C)CC1CCc1ccccc1 C(=O)(CCCc1ccsc1)NCC(C1CCC1)NC(CSCCN(C)C)=O C1(C#N)(C(=O)NC2(CC(=O)NC(c3ncnn3C)C)CC2)CC2CC2C1 C(=O)(C1=NOC(C)C1C)N1CCC(NC(c2c(CC)cccn2)=O)CC1C CC1CN(C(=O)CCCN2CCOC2=O)CC1(C)CNC(=O)C1=COCC1 N1(C(c2cnc(SC)[nH]2)=O)CC(NC(c2cc(C)n(C)n2)=O)C2CC12 c1(C(N2CCC(OC(C(N3CCC(C)C3)=O)C)CC2)=O)ccc2ncsc2c1 C1(CC)CN(C(C2CC(C3CCC3)C2)=O)CCC1NC(=O)CCc1cnoc1 c1(CC(=O)NCC(C(=O)OC)OC)cc(C=CC)ccc1OC(F)F N1(C(CN(C2CCCC2)C)=O)CC2(NC(C3CC4CC4C3)=O)CCCC2(F)C1 C1(CNC(CCS(C)=O)=O)CCC2CN(C(=O)CCCc3cc[nH]n3)CC12 c1(C(C(=O)NCC(C)(C)NC(=O)CC2COCC2O)O)ccc(F)c(F)c1 N1(C(C(C)Sc2ccccn2)=O)CC=C(CNC(=O)C2=CCSC2)CC1 c1(OC)ncnc(C(=O)N(CC(C)CNC(=O)C(C(C)C)SC)C)c1F c1(NC(C2(NC(=O)OC(C)(C)C)C(C)CCC2)=O)ccc(S(C)(=O)=O)[nH]1 C1(C(=O)NC2(CC=C)CN(C(c3ccc[nH]3)=O)C2)Cc2ccccc2CO1 C1(CCNC(CCN(C)CC)=O)CCCCN1C(c1c[nH]nc1OCCOC)=O c1(CCC(=O)NCC2CCC(NC(=O)Cc3ccns3)CC2)cc(F)cc(F)c1 CC1(C)COCC(CS(=O)(=O)NC(c2ccccc2Cl)CO)O1 c1(CCC)ccc(C(=O)NCC(O)CNC(C2CCC(O)C2)=O)s1 C#CCC(CC#C)C(=O)NC1CN(C(c2c[nH]nc2-n2cnnn2)=O)CC12CC2 C(=O)(C1=C(Cl)CCCC1)NCC1CN(C(COCCC#C)=O)CC12CC2 N1(C(=O)C2=CCCN(Cc3cccc(Br)n3)C2)CCn2c(Br)nnc2C1 C(=O)(C1=NOC(C)C1)NC(CN(C(c1c(C)cc[nH]1)=O)C)C c1(C(=O)NCC2C(NC(c3c(CC)cno3)=O)CC2)c[nH]c2nccc(Br)c12 C1(C(NOCCCC)=O)CN(C(=O)C(CC)CC)CCN1C(C)=O C1(C(N(C2CCOCC2)CCC)=O)CN(C(C2C3CC4C(C3=O)C24)=O)CC12CC2 C1(C(N2CC=CC(NC(=O)C(O)C(F)F)C2)=O)C2CCC3(COC(=O)C13)O2 CC12COC(C(=O)NCCCCNC(C3CC4CC4C3)=O)(C1)C2 CC1SCCCC1C(=O)NCCCCN(C(=O)C(C)(C)CO)C c1(C(N2CCC3C(NC(c4cnc(OCC)s4)=O)C32)=O)cc2ncccn2n1 c1(C(N(CCN(C(C(C)CF)=O)C)C)=O)ccc(Cc2ccccc2)cc1O c1(C(=O)OCC)cscc1NC(C1(NC(=O)COc2cccnc2)CC1)=O C(=O)(CC1=CC2CCC(C1)N2)NC(c1noc(C(C)(C)C)n1)C C(=O)(CCCN(C)N=O)N1CCCC(N(C(c2ccc(F)cc2N)=O)CC)CC1 c1(C(=O)NCCN(C(=O)CC2CCCC2(F)F)CCOC)cc(OC)ncn1 N1(C(C(CC)NC(N)=O)=O)CCC(c2cn(C(C)C)nn2)C12CC2 N1(C(C(CCC)OCC)=O)CC2(CCCC(CNC(c3cnsc3C)=O)O2)C1 C1(C(=O)NC2C(C)CN(C(=O)CCC3CCCCCC3)C2)C2CS(=O)(=O)CC12 C1(NC(C(COCC)C)=O)CC2CCC(C1)N2C(c1ccccc1SCCO)=O c1(CC)nn(C)cc1CNC(=O)C(C1CCCC1)NC(=O)C=Cc1nccs1 CC1CC(NC(CC(=O)NCCn2ccc(C(=O)O)n2)=O)CN1c1ncccn1 Cc1ccc(C(CO)NN(c2nccc(N3CCCCC3)n2)C2CC2)c(F)c1 N1(C(C(=O)NC(c2ccc(-n3ccnc3)cc2)C)=O)CCCC(CNC(N)=O)C1 C(=O)(CC(C)(C)C)N(CC(C)CNC(C1CN(c2ccccn2)C1)=O)C c1(C(=O)NCC2(OC)CCN(C(=O)Cn3cnnc3)C2)cc(P(C)(C)=O)cs1 CCCCC(C(=O)NCC1(O)CC(NC(c2ccc(F)cc2O)=O)C1)N(C)C c1(C(C(N2CC3(OCC(NC(CNC(C)=O)=O)C3)C2)=O)=O)c[nH]c2ccccc12 N1(C(C)=O)CCCC1C(=O)NCC1N(C(=O)C(C)CSc2ccccc2)CC1 c1(C(=O)NC2C(CC)N(C(=O)CCc3cccs3)CC2)cnc2sccc2c1 c1(C(=O)NC(CNC(C(CC=C)C(C)C)=O)C(C)C)c[nH]c2ccccc2c1=N CCC(C)(C)C(C)CC(=O)NC1CC2CCC1(NC(c1cc(C)c(C)nn1)=O)C2 Nc1cccc([N+](=O)[O-])c1C(N1C2CCC1CC(NC(=O)CNC=O)C2)=O c1(CC(=O)NCC(C)(C)NC(CSC)=O)ccc(NC(C)=O)cc1 C1(C(=O)NCCC(C)NC(c2cscc2Cl)=O)CNC(=O)N1C Cn1nc(Cl)c(C(=O)NC2CC(C)(NC(=O)Cc3ccc(Cl)cc3)C2)c1Cl C(C(=O)N1CCCC1CCNC(=O)C(C)(C)N(C)C)(C(C)(C)C)OC(C)(C)C N1(CCC(N2CCCCC2)C)C(=O)NC2(CCC(NC(C)(C)C)CC2)C1=O C(=O)(C#CC1(C)CC1)NCC1(C)N(C(C(C)NC(=O)NC)=O)CCC1 N1(C(C(C)N2CCC2)=O)CCC(CNC(C2OCC2(C)C)=O)C1 C(=O)(CS(=O)(=O)C1CC1)N1CC=C(CNC(C(C)(C)c2ccccc2)=O)CC1 CC(C)C(CNC(=O)C(C)Cc1ccco1)NC(C1(Nc2ccccc2)CC1)=O c1(C(=O)NC(CNC(C(C)=C2CCC2)=O)CC(F)(F)F)cc2nc(Cl)ccc2o1 c1(OC)cncc(C(=O)NCC23CC(CN2C(=O)CN2CCN(C)CC2)C3)c1C C1(C(=O)NCCC2(NC(=O)C=CC3CCC3)CCC2)CCCCC12CCC2 C(CCCCC(=O)NCCC(C)(C)NC(c1nc(C)n(-c2nc[nH]n2)n1)=O)SC C1(C(N2CCC(N(C(Cc3c(C)nsc3)=O)C)C2)=O)CCC(O)(C(F)(F)F)CC1 N#Cc1cccc([N+](=O)[O-])c1N1CCC2(NC(=O)CSC3CC3)CCCCCC12 C1(NC(c2cc(-c3ccc(C)o3)[nH]n2)=O)CN(C(C2CC(C)(F)C2)=O)CC1C O=C(CC1OCc2ccccc21)NC1CCN(C(=O)CCc2ncco2)C12CC2 C(CC(CC)C(=O)NC1CC1CNC(c1cncc(-n2cnnn2)c1)=O)=CC C(=O)(C1Cc2c(Cl)cccc21)N(C1CCN(C(c2c(C)occ2)=O)C1)C c1(C(N(CC(CNC(c2c(CC)occ2C)=O)C)C)=O)cnc(C)c(N)c1 c1(C(N2CC(CNC(Cc3cnc(C)[nH]3)=O)C(C)CC2)=O)ccc2nc[nH]c2n1 n1(CC)cc(Cl)c(C(N2CCCC(CN(C)C(c3cnn[nH]3)=O)C2)=O)n1 C(C)(C(=O)NNC(=O)COC(c1ccc2ncncc2c1)=O)SC c1(CNCc2cncc(OC)n2)ccc(F)c(F)c1O Cc1nc2cc(C(=O)NCC3CC3NC(=O)CC(O)CC(C)(C)C)ccc2o1 c1(CC(C(=O)OC(CC)CC#N)Sc2ccccc2Cl)ccc(F)cc1 c1(CSC)cccnc1C(=O)NC1CC1CNC(=O)Cc1csc(C)n1 Cc1csc(NC(C)C(=O)NCCCC(C)NC(=O)C(C2CCOCC2)C)n1 c1(C(N(CC(CN(C(=O)CC2(C)CCCC2)C)O)C)=O)ccc(N)cc1[N+](=O)[O-] c1(OCc2cc(C)no2)cc(C(C)C)n(C(C)(C)C)n1.c12ccc(cc1)c(=O)[nH]2 Cn1cc(OC2CCC2NC(=O)C(F)CC2CN(C(=O)OC(C)(C)C)C2)c(O)n1 N1(CCN2CCOCC2)CCC2CC2(NC(c2c(Cl)cn(C)n2)C2CC2)CC1 C1(Cn2cc(NC(C(COCC)n3cc(CO)nn3)=O)nn2)CC(O)C(O)C1 c1(C(C(=O)NCCN(CCCCCC)CCCC#C)OC)nccc2[nH]ccc12 CC1CCC=C1C(=O)N(C)CC1C2CN(C(=O)CSC(F)F)CC12 Cc1cc(C)cc(C=CC(=O)NCCS(=O)(=O)N2CCCC2)c1 Cc1c(C(N2CC(C(=O)NCC3CCCC(C)(C)O3)C(F)(F)C2)=O)cccc1F C(=O)(C(F)CC(C)(C)NC(=O)Cc1ccc(O)cc1)NC(C(CCC)C)CO C1(NC(CSCC(C)C)=O)CCC1CNC(C1(C2CCCO2)CC1)=O Cc1cccc(N(C)C(C2CC(F)CN(C(c3cc(I)ccc3O)=O)C2)=O)c1C O=C(C1=COCCC1)NC12CC(C1)N(C(=O)COc1ccc(F)c(Br)c1)C2 c1(CC(C)NC(C2OCCC2NC(=O)Cc2cnsc2)=O)ccncc1 C1(CNC(c2coc(Cl)c2)=O)CCCCN(C(C23CCC(F)(CC2)C3)=O)C1 c1(C(N(CC(=O)N(C)Cc2ncco2)C(C)C)=O)ncncc1N c1(NC(C2(C)CN(C(C3CCCCO3)=O)C2)=O)nc(Cl)c2c[nH]nc2n1 C(CCCC(CO)NC(=O)C#CC(C)(C)C)NC(C(CNC(C)=O)(C)C)=O c1(CC)cccc(CC(N2CCOC(C(C)NC(=O)C=C(Cl)Cl)C2)=O)c1 C(c1cncn1C)=CC(=O)NCC1CCN(C(C(C)C)=O)C1 N1(C(c2cc(C)ns2)=O)CCC(C(=O)N(C2CC2)C2CC2)(CF)C1 c1(CC(C(=O)N(C)C)N(C)C)ccc(F)cc1.c12csc(n1)CN(C=O)C2 c1(C(=O)NCC2(O)CCN(C(CC(CC)OC)=O)C2)cc2c(nc1N)CCCC2 C#CCC(C)C(=O)N1CCCC1CN(C)C(c1ncoc1-c1ccon1)=O c1(NC2CC(C)SC2)ccc(S(=O)(=O)NCCC(C)(C)C(F)(F)F)cc1C#N n1(CCCNC(C2CC(C)C(C)CC2)=O)cnc2ccc(F)cc2c1=O N1(C(CCNC(N)=O)=O)CCC(CNC(=O)C(C2CC2)C2CC2)CC1 C(C(F)C(=O)N1CC(C#N)C1)C1CN(C(CC2CN(C(C)=O)C2)=O)C1 c1(C(=O)NCCNC(c2c(C)c[nH]n2)=O)ccc(F)c(I)c1 C(=O)(C1Cc2ccccc21)N1CCC2CC(C(=O)NCCSCC)C2C1 N(C(=NCCc1ccccc1O)NCC1CCCCO1)C1C(COC)C1 C1(NC(C2CN(C(C3CCCO3)=O)CCO2)=O)CCCC2(CCC2)C1 C12(C(=O)Nc3cn(CC=C)nc3)CCCC1N(C(c1cc(OC)cs1)=O)CC2 N1(C(c2cnn(CCCC)c2C)=O)CCCC(NC(=O)CS(=O)(=O)NCC)CC1 CCC(O)C(C)C(=O)NC1CC2CC(NC(C3CC3(C)C)=O)C2C1 C1(CNC(C(C)NC(=O)NC)=O)CN(C(c2ccc(Cl)cc2)=O)CCCO1 C1(CCC)CN(N2CCC(c3nnc(C)o3)CC2)CCO1 c1(C(=O)NCC(C)(C)NC(c2cc(C)c(O)nn2)=O)ccc2ncccc2n1 N1(C(CNC(C)=O)=O)CCN(C(c2c(C)ccnc2C)=O)CC1CC(F)F c1(C(N2C(CCNC(c3ccc(F)nc3F)=O)CSCC2)=O)ncc(Cl)cc1Cl N1(C(C(C2CCOC2)OC)=O)CC(C)(CCC(=O)NCc2ccnn2C)C1 C1(C(N2CC3(CCCC3)C2)=O)(NC(CSCC)=O)CCC(C)(C)C1 Cc1cc(Br)c2[nH]c(CN3CC(Oc4ccccc4)C3)nc2c1 C#Cc1c[nH]nc1C(=O)N(C1(C(N2CCC2CC)=O)CC1)C CCCCCCCCCS(=O)(=O)N1CC2OC(C)(C)OC2C1 C(C(C)(C)CNC(=O)CC1CCCC1NC(=O)CN1CCCC1)OC C1(CCC)C(C)CCCN1C(=O)C=CCN(C)C(c1ccc(C)c(O)c1)=O N#Cc1ccc(C=CC(=O)NCC2CC(NC(C34CCC(CC3)CC4)=O)C2)cc1 FC1(F)Oc2cccc(CNCC3CC34CCOC4)c2O1 C1(C)(C(=O)NCCOC2CCN(C(C(C#C)(C)C)=O)C2)CCCCNC1=O c1(-n2cc(C(C(C)(C)C)NC(C3CC3C(=O)O)=O)nn2)ccc(CO)cc1 C1(NC(CNC(=O)NC)=O)CCN(C(=O)CCCCCc2cccs2)CC1O Cc1cc(C(=O)NC2(C(F)F)CC(F)(F)C2)c(F)c(Br)c1 C1(NC(C=C(CC)CC)=O)CN(C(=O)C(C)=CC2CC2)CC1c1ccccc1 c1(NC(=O)NCCS(=NC)(C)=O)ccc(Cl)c(OC)c1 N1(C(CCCCCCCC)=O)CCC2CCN(C(=O)COCC(F)F)CC2C1 n1(CCC(=O)NC(CNC(C=C(C)C(F)F)=O)C)nc(C)c([N+](=O)[O-])c1C c1(OCC)ccc2cc(C(c3nnnn3C)NC3(CF)CCC3)oc2c1 C1(C)(CNC(C2(C)CCSCC2)=O)COCCN(C(C2CC(F)(F)C2)=O)C1 Cc1nc(N2CC3CC2C3C(N2CCC(CN(C)C)CC2)=O)c2c[nH]nc2n1 N1(C(C2N(C(=O)OCC)CSC2)=O)CCOCC1CNC(=O)C(C)(C)F [N-]=[N+]=NC1CCC(C(=O)NCC(C2CC2)NC(=O)CNC(N)=O)CC1 Cc1ccc(N2CCC(NC(=NCC3CCS(=O)(=O)N3)Nc3cccs3)C2)cc1 C1(CC)(NC(C2CC3C=CC2O3)=O)CCN(C(=O)CCc2csnn2)CC1 Cc1ccc(C(N2CCC3(CC3C(=O)NC(C)(C)CC(C)(C)C)C2)=O)c(F)c1 Cc1cc(C(=O)NCC2CN(C(=O)CN(C3CCC3)C)CCN2C)ccc1O CC1CN(C(c2ccc(Cl)cc2)=O)CC(C(=O)NOCC2CC2)O1 C1(C2CCCCC2)(NC(C2N(C(CSC(C)(C)C)=O)CC(O)CC2)=O)CC1 Cc1ccc(F)c(C(=O)NCC2CCCN2C(=O)C(C)OCCC(C)C)c1 N1(C(c2ccc(C)nc2O)=O)CCC2CC(NC(=O)C3=COCCC3)CCC2C1 C=CC1CCN(C(C2CCCC2CNC(c2ncn(CC)n2)=O)=O)CC1 c1(NC)c(C(=O)NC2CC(F)(CNC(=O)CN3C(=O)CCC3=O)C2)cccc1F C(=O)(CC(O)(CC)c1ccccc1)NCCCNC(COCC)=O c1(C(N2C(CNC(c3c(SC)cccc3)=O)C(C)CC2)=O)cn(C)c(=O)cn1 CC(C)(C(=O)N1CC2C(NC(=O)C(O)C3=CCCCC3)C2C1)S(=O)(=O)C1CC1 CCC(CC)=CC(=O)NC(CNC(C1CC(C(F)F)C1)=O)CO C(=O)(C1=CCc2ccccc21)NC1CCCN(C(c2ccc(C(=O)OC)[nH]2)=O)C1 C1(C(=O)NC(c2ccncn2)C)CC2(CCC2)CN1C(=O)CC1=CCCCC1 C(CCC(c1ccccc1)NC(=O)CSCCC(F)(F)F)NC(C(C)OC)=O S(=O)(=O)(CCC(=O)NCCC1CCCCN1C(=O)Cc1ccc(O)cc1)N(C)C CCCCC(C(=O)N(C)CCN(C(=O)C(F)(F)CC1CCCO1)C)C(C)C C(=O)(CCCC(C)(C)C(=O)OC)N1CC2C(N(C(C3N(CC)CCC3)=O)C)C2C1 CN1CC(F)CC1C(N1CC(O)(CCNC(c2cccc[n+]2[O-])=O)C1)=O C1(OC)CC2CC1CN(C(C1CCOCC1NC(c1ccn(C)c(=O)c1)=O)=O)C2 c1(CC)cc(C(=O)NC(C(C)NC(=O)CC(=O)N(C)C)C(C)C)ccn1 c1(CNC(C(C2CCCOC2)N(CC(=O)NC)CC)=O)nnn(C)n1 CC1CCCCN1CC(N1CC(F)CC1CC(=O)NC1(C(C)O)CC1)=O C1(OC)CCCN(C(=O)C(CC2CCC2)NC(=O)C(F)=CC2CC2)C1 N1(c2ccnc(COC)n2)CCCC2(NC(c3cccn(C)c3=O)=O)CCCC12 n1(CC(=O)N(CCN(C(C2(CC#C)CCCCC2)=O)C)C)ccc(=O)c(O)c1C O=C1CC(CC(N2CC(NC(=O)CSc3ccncc3)C2)=O)CCN1 N1(C(C2CN(C)C2)=O)CCC2(CC1)CN(Cc1cscn1)C2 C(=O)(CCS(N)(=O)=O)NC(C(=O)NCC1C(N(C)C)CCC1)C1(O)CCC1 C1(CNC(C(COC)(F)F)=O)CC(C(F)(F)F)CCN1C(=O)C=C1CCN(C)C1 C=CC1(C(N2CCC(C(=O)OCC)C2)=O)CCN(C(=O)C(C)N2CCCC2)C1 c1(CNC(C2(C(C)=O)CC2)=O)ccc(CNC(C2C3CCCCC23)=O)cc1F C(=O)(C(C#N)C(C)(C)C)N1CC(CN(C(c2c(OC(C)C)n[nH]c2)=O)C)OCC1 CC1(C)CN(C(=O)C2=CCN(C(=O)Cc3cccnc3)C2)CC(=O)N1 N1(C(Cc2ccc(C)s2)=O)CCN(CCNC(C2C(C)(C)C2(F)F)=O)CC1 C1(NC(c2c(CC=C)cccc2)=O)CCCCCN(C(=O)C=C(C)C(F)F)C1 c1(C(=O)OC)ccc(NC(C2COCCN2Cc2cc(Cl)nc(Cl)c2)=O)cc1Br c1(NC(=O)N(C2CCNCC23CC3)CC23CCN(CC2)C3)ncnc2c1CCC2 C=Cc1cncc(C(=O)NCc2ccc(C(=O)NCC(CN(C)C)OC)cc2)c1 C1(C(C)C)N(C(C2CC=CC2)=O)CC12CCN(C(C1CC(C)(C)CO1)=O)CC2 N1(C(c2c(O)nc(CC)c(C)c2)=O)CCC2CCN(C(c3csnn3)=O)C2C1 C#Cc1cccc(C(N2CC3CC(C2)C3NC(=O)CC2CCC(=O)NC2)=O)c1F C(C)(CC(F)(F)F)NC(COC1CN(C(Cc2nc(C)[nH]n2)=O)C1)=O c1(OC)cc(NC(C2CCC(NC(c3cc(Cl)ccc3Br)=O)C2)=O)c(Br)cc1C Cc1ccc(Br)c(C(=O)NC(CNC(=O)Cc2cc[nH]c(=N)c2)CO)c1F O=C(C1=NOC(c2ccccc2)C1)NCC1CN(C(C2CN3CCCC2C3)=O)C1 Fc1cccc2c(=NC(CN3CCCC3)CC3CC3)[nH]c(=NCc3cncs3)[nH]c12 c1(C(N(CC(C)NC(C2(CO)CC2(F)F)=O)C)=O)c[nH]ccc1=N C1(CC(=O)N(CC(C)C#N)C)(OC)CN(C(=O)CCC2CCC(=O)C2)C1 N1(C(c2c(C)cn(C)c2)=O)CCN(C(=O)CCC(C)N(C)C)C2CCCC2(C)C1 c1(C(=O)NC2CN(C(C(C3CCCCC3)OC)=O)C(C)C2)ccc2c(c1)OCO2 C1(C(=O)NC(=O)OC(C)(C)C)CC(C(N2CCC(c3cc[nH]c3)CC2)=O)CC1O C1(NC(CN2CCC(C)CC2)=O)CC2(CCN(C(=O)CC3CCS(=O)(=O)C3)C2)C1 C1(C(=O)NCC2(CNC(CN(C)CC)=O)CC2(F)F)CC(C)CC(=O)N1 c1(C(N(C2CCN(C(C(CC)C)=O)C2)C)=O)nc2ccccc2s1 c1(OC)cccc2c1OCCCC2NC(c1cc(Br)c(Br)[nH]1)=O c1(CC)sc(C(=O)NC2CCN(C(=O)C(c3ccccc3)NC(C)=O)C2)cc1C c1(C(=O)NCCC(C)(C)NC(c2cocn2)=O)c(Br)nc2n1CCCC2 c1(CC(=O)NCCN(C(C=CSC)=O)C)c[nH]c2nccc(Cl)c12 C1(CCNC(c2ocnc2C(F)F)=O)CCC(NC(=O)C(O)C2CCC2)C1 c1(C(C)(C)C)conc1C(=O)NC1CCC(NC(=O)Cc2cccs2)C1 C1(N(C(=O)CCC2CCN(C(c3cnsc3)=O)C2)CC)CCC(O)CC1 O(NC(=O)CCC(C)(C)[N+](=O)[O-])C(C(=O)ON1CC=CC(CC)C1)CC(C)C c1(OC)nn(C)c(Br)c1C(=O)NCC1CC1NC(c1c[nH]nc1C)=O CCCCCCC(=O)N1CC(N(C)C(c2coc(C(F)(F)F)c2)=O)C(O)C1 C(=O)(C(C)(C)C(C)(C)O)NCC=CCC(=O)NCC1CCCC(C)O1 C12(C(=O)NC(CC)CNC(C3(n4cnnn4)CC3)=O)CC(C#N)(C1)C2 C(=O)(C1=NN(CCO)C(=O)CC1)N1CCN(C(CC2CC(C)C2)=O)CC1CCO N1(C(CCOC)=O)CC(O)CC1CNC(c1cnc(-c2ccccc2)nc1)=O c1(C(=O)NCC2(C)CCCS2)c(Cl)cccc1I C1(NC(c2csnn2)=O)CC2CCC1N2C(c1cncc(Cl)c1Cl)=O c1(CC)nc(C)c(C(N2CCC(C)C2CNC(=O)C(c2nc(C)cs2)C)=O)s1 N1(C(C2(C)COC2)=O)CCCC(C(=O)NC2(CF)CC2)C1 CCCC(C)(O)CC(=O)NC(c1ccnn1C)C(=O)NC1(C)CC=CCC1 C1(CCC(=O)N(CC(CN(C(CCCOC(C)C)=O)C)O)C)CCCCN1C C1(CC(=O)NC(C)C(CO)NC(C2CC(O)C2)=O)CC2(CC2)CO1 c1(CC(N2CCC(CNC(c3c[nH]nc3F)=O)C2)=O)csc2c(Cl)cccc12 c1(CCC)noc(CCCC(=O)NCC(CC)NC(C2CC(C)CO2)=O)n1 c1(C(C)C)ccc(OCCC(=O)NC2(C)CN(C(=O)CN3CC(C)C3)C2)cc1 C(=O)(C1CCc2c[nH]nc21)NCC(CC(C)C)NC(C(C)OC)=O c1(C(c2nnnn2C(C)C)NC(CC)C2CC2)c(F)cc(F)c(Br)c1F C(=O)(C(O)CCCNC(C1(C#N)CCOCC1)=O)NC1C(C)CCC1C c1(C(N2CCCCC2c2cn[nH]c2)C(=O)NC(CC)C)ccc(C)c(Br)c1C CCC(CC)CC(=O)N1CCCC(O)(CNC(C23CCCC2(C(N)=O)C3)=O)C1 CC(C)(C#N)CCC(=O)N1CC(c2ccccc2)(NC(=O)CC2CC2)C1 c1(OC)cc(C)ccc1C(=O)NCC(CO)NC(=O)CC(=O)OCCC(C)C c1(CC(C)C(=O)NCC(C(C)(F)F)c2ccccc2)ccc(N)cc1 C1(CNC(C2CC(C(F)F)C2)=O)CN(C(C2CCC2)=O)CCC1(F)F C1(NC(C(CC2CCC2)OC)=O)COC2CN(C(=O)CNC(N)=O)CC12 c1(CCC(=O)NC2C(N(C(=O)CCC3CC3)C)CCCC2)cnc2n1CCOC2 C12(NC(C3(OCC)CCC3)=O)CCCC(CN(C(c3ccco3)=O)C1)C2 c1(C(=O)NCC(CN(C(CSCCC)=O)C)C)c(C)c2ccc(F)cc2oc1=O Clc1nc(C2CCC2)cc(=NCC2CCC(C3CC3)O2)[nH]1 C(=O)(CC(C)(O)C=C)NC1(C(N2CCC(OCC#C)CC2)=O)CC1 N1(C(CN(CC)CC2CCCC2)=O)CCC(C)C(N(c2cc(=O)n(C)cn2)C)C1 N1(CCC(=O)N(C)CC2CCN(C(Cn3ccc(C)n3)=O)C2)CCCCC1=O C1(C(=O)NC(CC(C)C)(C)CNC(=O)CCC(N)=O)Cc2cccnc2C1 c1(C(=O)NC(CC)C(OC)OC)nc(C)n(-c2ccc(Cl)cc2)n1 N1(C(=O)OC)CCCC(CNC(=O)NC2CN(C)CCO2)C1 c1(CC(N2CCOC(C3CCCOC3)C2)=O)ccc(Br)c(Cl)c1F Cc1cc(F)cc(C#N)c1S(=O)(=O)N1CC(C)(CS(C)(=O)=O)C1 c1(C(=O)NC(CNC(=O)CCc2cscn2)C2CC2)cc2sccc2s1 c1(CNC(CC2N(C)CCC2)=O)cccc(NC(=O)CCc2cc(Cl)cs2)c1 C1(CNC(Cc2c(C)n[nH]c2)=O)COCCN(C(C2CCCCC2)=O)C1 C#CCC(C(=O)N1CCC1(C)CCC)NC(=O)Cc1cc(C)n(C)n1 N1(C(C(CN(C)C)O)=O)CCC(NC(C2CCOC2)=O)C(C(N)=O)C1 N1(C(C2C(C(=O)OCC)C3C2CC3)=O)CC2CC(NC(c3cocn3)=O)C1C2 CCC(C(=O)OC)C(=O)NCC1CN(C(C2CCC(O)CN2C)=O)C1 c1(C(=O)NC2CN(C(C3CC(C(F)(F)F)CO3)=O)C2)ccnc(C(N)=O)c1 N1(C(c2c(CNC(c3ccc(C)c(C)n3)=O)cco2)=O)CCSC2CCCC12 C1(C(N(C)CC2(n3ccc(C4CC4)n3)CC2)=O)C2CC3C(C2)C13 N1(C(c2c(CC)n[nH]c2)=O)CC2CN(C(C3(OC)CCCSC3)=O)CC2(C)C1 C(C(=O)N1CC2C(C(=O)Nc3cnn(C(C)C)c3)C2C1)(C(C)C)OC N1(C(c2cc(C)c(C)s2)=O)C2CCC1CC(NC(=O)C(C)C(O)C(C)C)C2 c1(CCC(=O)NC23CC(C(=O)Nc4cn(CC)nc4)(C2)C3)nc2ccccc2o1 c1(C(=O)NC2CN(C(C=C(CC)C)=O)CC(C)C2)cccc2cccc(C)c12 c1(C(N2C(CNC(CCC=CCC=C)=O)CC(O)C2)=O)cncc2sccc12 Clc1cc(Br)ccc1CNC(c1cncnc1)c1nnnn1C1COC1 N1(C(C=Cc2cc(C)no2)=O)CCCCC(C(=O)NCc2ncc(C)o2)C1 C#CC1CN(C(c2cc([N+](=O)[O-])n[nH]2)=O)CCN1C(C1CC1C(C)C)=O C1(C2CN(C(=O)C(c3cnn(C)c3)O)C2)(NC(C(c2ccc(CC)s2)=O)=O)CC1 c1(CC(=O)N(C2CCN(C(C3CC(N(C)C)C3)=O)C2)CCC)cnccc1C N1(C(C(COCC)Oc2cncs2)=O)CCCC(C(=O)NCCO)C1 c1(CC)ccc(Br)cc1NC(C)Cc1cccc(Br)c1 c1(NC(c2nc(C)[nH]n2)C)nccc(=NC2CC3(CCC3O)C2)[nH]1 N1(C(C(=O)NCC)=O)CCN(C(=O)C(O)CC2CCOCC2)CC2CCCCC12 CC(C)CC(C)C(=O)N(CC(O)CN(C)Cc1cc(O)ccc1Cl)C C1(NC(CNC(N)=O)=O)CCCC1CNC(=O)CCc1nnc(C2CCCC2)o1 C1(CNC(c2c(CC)cccc2)=O)N(C(C2COC(=O)N2)=O)CCCC1(C)C C1(C(N(C)CCNC(C2(c3ccno3)CCC2)=O)=O)C2CS(=O)(=O)CC12 CC(=Cn1ccnn1)C(=O)N1CC=CC(NC(=O)C2=CCSC2)C1 CN1CCC(F)(C(N2CCC(C)(CNC(C3CC(C4CC4)=NO3)=O)C2)=O)CC1 N1(C(c2cc(COC)no2)=O)CC(CNC(C2(C(F)(F)F)CCC2)=O)C(O)C1 C(=O)(C(C)(C)C(=O)N(C1CC1)CC)N[SH](=NCC)=O C1(CC(=O)NCC(C)C#N)CC2(C1)CN(C(C1(C(F)(F)F)CC1)=O)C2 N1(C(C(N2CCOCC2)C)=O)CCCC1CNC(=O)CCN1CCC1 C1(C(N(C2CC(F)(F)C2)C)=O)CCN(C(=O)C(F)n2ccnc2)C(C)(C)C1 N1(C(C(CC)NC(C)=O)=O)CCCC(C(=O)NCCCc2cccc(C)c2)CC1 c1(OC)ccc2nc(NC(=O)CSCc3c(I)cnn3C)[nH]c2c1 c1(C(=O)NCCC2OCCCN(C(COCC)=O)C2)cnc2n1CCCC2 C1(NC(COCC(C)(C)C)=O)CC12CC(NC(c1ccccc1)=O)C2 C1(CC)CCN(C(=O)CC2CCCCC2NC(c2cc(CO)n(C)n2)=O)CC1 C(C1CC1)(C1CC1)=CC(=O)NCCC1(C(=O)NC2(C)CC(O)C2)CCC1 c1(C(=O)NC2C(CNC(C=CC(=O)N(C)C)=O)CCC2)c(F)ccc(F)c1O c1(SCOC(N2CCCCC2C2(O)CC2)=O)nc2ccc(C(=O)O)cc2s1 c1(C(N2CCC(NC(C3(C)CC(C#N)C3)=O)C(CO)C2)=O)ccc2cnnn2c1 C1(C(=O)NCC(C)(C)CNC(=O)Cn2nnc(=O)[nH]2)(OC)CCOC1 c1(CCC(=O)NC2CCN(C(C3CCSC3)=O)CC2F)ccc2c(c1)OCCO2 CC1OC(=O)NC1C(N1CCC(C(N2CC(CC3CC3)C2)=O)C1C)=O c1(C(=O)NCC(CC)NC(=O)C(C(C)O)N(C)C)nc(C)[nH]c1C(F)(F)F c1(CNC(C(COC)OC)=O)cc2n(n1)CCN(C(C1CC1C1CC1)=O)C2 C(=O)(CCC(C)CN(C)C)NCCCOC1CCN(C(C(CC)(C)O)=O)CC1 C(=O)(CC1=CCCC1)N1CCC(CC=C)(C(N2CCC(=C)CC2)=O)C1 c1(CC)ccc(C(=O)N(C)CC2CCN(C(=O)C(C)(O)CC)C2)cc1Br c1(C(=O)NCC2N(C(C3(C)C(C)CCC3)=O)CCC2)cnc2c(c1)CCOC2 Cc1cc(C(N2CCC(CNC(=O)CCC(C)N(C)C)C2)=O)ccc1Cl C1(C(N(CC)CC2CCNC2=O)=O)CCN(C(C)CCO)CC1 CN1CCc2cc(C(=O)NC3CCOCC3NC(c3ccco3)=O)ccc21 c1(CNC(c2cccc(-c3n(CC)nnn3)c2)=O)ncc(F)cc1F CC(C)(C)C#CC(=O)NCCC(O)CNC(=O)Cc1csc(NC=O)n1 C=CC(C)(O)CCCC(C)C(=O)NCc1ccnc(-c2ccccc2)c1 C1(NC(C(COC)(C)OC)=O)CN(C(=O)C2=NOCC2)CCC1C(F)(F)F N1(C(c2ccc(OCCCl)cc2)C(=O)NCCC#N)CCC2(CCCOC2)CC1 S(=O)(=O)(c1ccc(Br)cc1NCc1cc2sccc2s1)N1CC(C(C)C)SCC1 O=C(CCN=c1cccc(S(=O)(=O)NCCC2OCCCO2)[nH]1)NC1CC1 C1(C(=O)NCC(=O)NCC=C)CCN(C(C2CCSC2)=O)C(C)(C)C1 N1(C(CCC2CC(C)C2)=O)CC(C(=O)NC(C(C)(C)O)C2CC2)C(F)(F)C1 C(=O)(C(C)(COC)CC)N1CCCC(CN(C(CCNS(CC)(=O)=O)=O)C)C1 C1(NC(c2c(C)ccc(OC)c2)=O)CN(C(=O)C(C)SC)C2CCCC12 N1(C(C(C)(Cl)Cl)=O)CC(c2cn(CC(O)C(F)(F)F)nn2)C(C)(C)C1 C1(COC)CC(CNC(c2cnc(C)cn2)=O)N(C(c2nc(C3CC3)cs2)=O)C1 N1(C(c2nc(C)sc2Br)=O)C2CCC1C(CNC(=O)C(C)C1CC1)C2 N1(C(C(CC#C)O)=O)CCN(C(c2cncc(O)c2Cl)=O)C2COCC12 C1(C(N2CCC(c3c(CNC(C(C=C)(C)C)=O)c[nH]n3)C2)=O)CC2C(C1)C2(F)F c1(CC(=O)NC(C2OCCN(C(c3cc(C)[nH]c3)=O)C2)C)ccc(O)c(O)c1 C1(S(C)(=O)=O)(C(N2CC(C(C)NC(=O)CC3CCC4CC34)C2)=O)CCCC1 CC1OCCC1C(N1CC(CC(C)NC(c2sccc2OC(C)(C)C)=O)C1)=O CC1(C(=O)Nc2cc(-c3ccccc3)no2)CCCN1Cc1ccc(Br)[nH]1 c1(C(=O)NC23CCCN(C(C(CCCC)O)=O)CC2C3)nc(C)n2ccccc12 c1(OC)ccc(C(N2C3CCC2CC(CNC(=O)CC2CC2C)C3)=O)c(F)c1N N1(C(C2(CC(C)C)COC2)=O)C2CCC1C(F)C(NC(=O)CC(C)P(C)(C)=O)C2 N1(C(c2c(C)con2)=O)CC(NC(c2c(C)nsc2Br)=O)C(C)(C)C1 C(CNC(C12CC(CC(F)F)(C1)C2)=O)(CCNC(C1(N(C)C)CCCC1)=O)OC c1(C(N(CCC(C)NC(C(c2ccccc2)OC)=O)C)=O)c(C)ccc(F)c1N C1(O)(C(=O)NCC2CCC(NC(C#CC)=O)C2)CCCN(C(=O)OC(C)(C)C)C1 C(=O)(C(O)CCC(C)C)NCC(C(=O)N(CC#CC)CC#C)O c1(NC(CC2CN(C(c3c(C)nc(C)o3)=O)CC2C)=O)cc(C)c(O)cc1C c1(CC(N2C(C)(C(=O)OC)CC2)=O)ccc2c(c1)CCCS2(=O)=O C1(C(=O)NCCN(C(C2N(C)CC(F)C2)=O)CCOCCO)CCOCC1(C)C c1(OCC(=O)NCC(CO)NC(c2c(C)c[nH]n2)=O)cccc(S(C)(=O)=O)c1 C1(C(=O)OC)CCC(C)N(C(c2cc(C)oc2C)C(=O)NCCCF)C1 CCCCCC(O)CC(=O)NCCc1ocnc1CNC(c1ccncc1C)=O Cc1ccc(C=CC(=O)NCC2CCCN2C(=O)CC2CC(C(F)F)C2)o1 N1(C(c2[nH]cc(C(C)=O)c2)=O)CCC=CC1C(=O)NC1CCCC1(F)F c1(C(N2CC(C(N(CCCO)CCC)=O)(CC)C2)=O)ncccc1C Cc1cnc(C(N2CCCC(C(C)NC(c3ccc(O)nc3C)=O)C2)=O)cc1Cl Cc1cccc2cc(C(=O)NC(CNc3ncc(Br)c(O)n3)C(C)(C)C)nn12 C1(NC(CSC)=O)CC2CN(C(=O)CCCNC(=O)NCO)CC12 N1(C(C=COCC)=O)CCCC2CN(C(c3c(C)nc(C)n3O)=O)CCC12 c1(CC(C(=O)O)NC(c2c(C(C)C)c(Br)ccc2)=O)cnc2ccccc2c1 Cn1cc(S(N)(=O)=O)cc1C(=O)C(=O)Nc1cn(C)nc1CN1CCCC1 N1(C(c2cnn3c2CCC3)C(=O)NCCCOC)CCC2(CC1)CC(OC)C2 c1(OC)oc(C)nc1C(=O)NC(C)(CNC(c1nc(Cl)sc1Cl)=O)C(C)C N1(C(C(CC)(F)C(=O)OC)=O)CCC2CCC(C1)N2C(=O)CCn1cc(C)cn1 N1(C(c2c(C)[nH]nc2CO)=O)CC2(CCC(NC(C3CC3(C)C)=O)CC2)C1 c1(NCCOC)cc2c(cc1OC)CCCC2 CCC(CC)C(C)C(=O)N1CCN(C(=O)CC(C)(C)O)C(CC(F)(F)F)C1 c1(SC)ncc(C(N2CCC(CNC(C3COCCN3C)=O)C(C)C2)=O)c(O)n1 c12cc3c(cc1Br)CCN(C3)C2.c1(-c2c(CO)c[nH]n2)cccc(C(F)(F)F)c1 c1(CC)sc(=N)[nH]c1C(=O)NCCN(C(c1coc(Br)c1)=O)CC c1(C(C)=O)cc(NCCC2CC(NC(C3(C)CC3(F)Cl)=O)C2)ccc1[N+](=O)[O-] N1(Cc2ccc(-c3c(N(C)C)cccc3)cn2)CCc2ncncc2C1 C(CCCCCN(C(=O)CCCCO)C)NC(CN(C)CCNC(=O)CCS(C)=O)=O CCC(C(=O)NCCCCC(CO)NC(c1cncc(C)c1)=O)C(F)(F)F N1(C(c2c(=N)cc[nH]c2)=O)CCC2(CCCC2C(N2CCSCC2CO)=O)C1 C(=O)(C#CC1CCN1NC(=O)OC(C)(C)C)NC(C1CN(C)CCO1)C c1(CSc2cccc(C(=O)OCC)c2)nc(Cl)ccc1N c1(C(=O)NC2C(NC(C3(CC=C)CC3)=O)CC2)cc(Cl)c(Cl)c([N+](=O)[O-])c1 C(=O)(C1=C(C)CCOC1)N(CC(CO)(CO)NC(CC1(C=C)CCC1)=O)CC S(=O)(=O)(c1ccc(Br)cc1F)NC1C(C(=O)NCc2cc(C)nn2C)C1 C1(C(=O)NCC2NC(=O)OC2)COCCN1C(=O)CCCn1cncn1 CN1CCC(C(N2CC(O)CC2C(=O)NCC2(C)CSC2)=O)CC1=O c1(COCC(=O)NCCN(C(C(C2CCCOC2)OCC)=O)C)ccccc1Cl C(=O)(CC(F)(F)C(F)(F)F)N(C)CC1(O)CCN(C(c2ccoc2)=O)CC1 N1(C(C(C)(C)Cl)=O)CCC(C)(C)C(C(N2CC(C3CCCO3)C2)=O)C1 C(=O)(CCCC(C)(C)C#N)N(C(CC)CC(=O)NCC1CC(NC)C1)C N1(C(c2n(CC)ncc2)=O)CCN(C(c2coc(O)n2)=O)C(CC(F)(F)F)C1 Cc1cc(C(=O)NC2CCC2NC(=O)CCC2CCCC(=O)N2)c(C)[nH]1 c1(C(C)C(N2CCN(C(C3CCC(C)O3)=O)CC2C)=O)cn(C)c2ccccc12 CCC(CC(F)F)C(=O)NC1CC12CCN(C(=O)Cc1ccccc1)CC2 C(O)(C(=O)N1CC=CCO1)C1CCN(C(CC2(C#N)CC2)=O)C1 C(=O)(CCC(C)(C)C(=O)N1CCC(N(C)C(c2coc(C(F)(F)F)n2)=O)C1)OC c1(CC)n[nH]cc1C(N1CCC(OCC(C)C)C1)C(=O)NC1CCCC1 Cc1ccc(C=CC(=O)N(CCCO)C(C)(C)C)cc1C N1(C(CC2(N(C)C)CC2)=O)CC2CC1C2C(=O)NC1CC1F Cn1ncc2cc(-c3c[nH]nc3C(=O)NCCc3nccs3)ccc12 CCCC(C(=O)NCC(CNC(c1cc(C(C)(C)C)c[nH]1)=O)CO)N(C)C CN1CCCC1CCNC(=O)C(C1(O)CCC1)NC(=O)CCc1nncs1 Cc1cc(S(C)(=O)=O)cc(C(N2CCN(C(=O)CCCN=[N+]=[N-])C3CC23)=O)c1C c1(C(N2CCC(NC(CC(CC)C3CCC3)=O)C2C)=O)cnc2cc[nH]c2c1 Cc1cc(C(=O)NC(C2CCCCN2C(=O)C=C2CC2)C)c2sc(=N)[nH]c2n1 CC1(NC(c2nccnc2Cl)=O)CCCN(C(=O)C(O)CC2CCCCC2)C1 C(=O)(CC(C)CNC(=O)CC1C=CCC1)N(CCCOC)C C(=O)(CC(C)P(C)(C)=O)NCC1(NC(c2c(C)nc(CO)o2)=O)CCC1 C1(C(N2CCSCC2c2ccccc2)=O)CCCCN1S(=O)(=O)CCCCl Cc1nsc(C(=O)NCC2CCN(C(C3(n4cnnn4)CCOCC3)=O)C2)c1N CCC(C)CC(C(=O)NCCC(C)(C)O)NC(C1CCN1C)=O C12(CCCCCC1)CO2.c1(C(=O)NCCOCC(=O)OC)ccc(CSC)cc1 Cn1cc2cc(CC(=O)NCC3(NC(=O)C4=COCCO4)CCOC3)ccc2n1 CCCCC(C(=O)NCCC1(CO)CCC1)NC(C1CC2CC2C1)=O CCS(C)(=O)=NC(=O)CC(c1ccccc1Cl)N(C)C c1(C(N(CCNC(C2CC(OC)C(OC)C2)=O)CC2CC2)=O)cccc2scnc12 c1(C2(CNCC(=O)NC(C(=O)OC)C)CCC2)ccc(Br)c(C)c1 N1(C(CC(c2ccc(F)cc2F)NC(C(CC)C)=O)=O)CCCN(CC#N)CC1 CC(CC(=O)NCCCCC1CN(C(=O)C=CCF)C1)n1cc(Br)cn1 c1(C(=O)NC(C(C)NC(c2ccc(CC)o2)=O)C)cc(C)n(C)n1 c1(CC)ccc(S(=O)(=O)N2CC3C(NCc4c(Br)ccc(F)c4F)C3C2)cc1 CC1CN(C(c2coc(C3CCCCC3)n2)=O)CC1Nc1ncc(I)cn1 C12(CSC3CN(C(CC(C)N4CCCC4)=O)C(=O)C3)CCC(CC1O)C2 C1(NC(C(F)=CCC)=O)CN(C(C2CC(SC)C2)=O)CC12CCC2 c1(CC)nc(C)[nH]c1C(=O)N(CCCN(C(=O)CCCNS(C)(=O)=O)C)C C1(NC(CSCC=C)=O)CC(C)N(C(c2ccc(-c3csc(C)n3)s2)=O)C1 N1(C(C2=C(C)OCC2)=O)CC2CCC1C(NC(=O)CC1(CO)CCOCC1)C2 CCCCC(O)C(=O)NCCC1CC(NC(c2cc3n(n2)CCC3)=O)C1 C(C(C)(C(=O)NCCCN(C(=O)CC1CCOCC1)C(C)C)OC)OC C#CCC(C)(C)C(=O)N1CCOC(C(C)NC(c2snc(O)c2Cl)=O)C1 C(=O)(C(CC(C)C)CC(C)C)N1CC2CCN(C(c3c(C)ccs3)=O)CC21 c1(C(=O)NCC2(N(C(C3(CCl)CCC3)=O)CCO)CCC2)cc2scnc2[nH]1 c1(SC)nc(C)cc(=NC2CN(C(=O)C(C)(C)CC(C)C)CC3(CCC3)C2)[nH]1 C=C1Cn2c(C(=O)NC3(CO)CN(C(=O)CC4C=CCCC4)C3)nnc2S1 CC1CCCC(CN2CCN(C(CNc3ccc(CS(C)(=O)=O)cc3)=O)CC2)C1 C(=O)(C#CC1CCCCC1)NC(C(=O)NCc1[nH]nc(C(C)C)n1)c1ccco1 [N-]=[N+]=NCCCCCCC(=O)NC1(CNC(c2csc(-c3nc[nH]n3)n2)=O)CC1 C1(O)(CN(C(c2c(CC)nns2)=O)C)CCCN(C(c2cc(C3CC3)[nH]n2)=O)C1 C=C(C)C1CN(C(c2c[nH]nc2CCNC(c2nn(C)cc2C)=O)=O)CCO1 Cc1cc(F)ccc1C1(C(N2CC3C(CNC(=O)CCC4CC(C)C4)C3C2)=O)CC1 C1C(F)(C(C)C)C(=O)N2CC(C2)C(=O)N1.C1(OC)CCN(CC(=O)N(C)C)C1 N12CCC13CN(C3)Cc1ccc(cc1)OCC2=O.c1(C(=O)OC)ccncc1 c1(C(N2CC(NC(CC=CCC)=O)C3C2C3)=O)ccc(-c2ccco2)nc1O c1(C(=O)NCC2N(C(Cc3c(C)non3)=O)CC(C)CC2)ccn2nncc2c1 Cc1cc(C(N2CC(O)(C3CCCN3C(c3cccnc3O)=O)C2)=O)c(C)c(C)c1 N1(C(CSC2N(C(CC(C)C)=O)CC=C2)=O)CCC(O)(c2ccccc2)CC1 CC1CN(C(c2ccc(C(F)F)o2)=O)CCC1NC(=O)CCOc1cccnc1 Cc1cc(C(=O)N(C)CC2COCCN2C(=O)Cc2ccsc2Cl)nnc1O CC1CN(C(C23C(NC(=O)CNC(C4CC4C)=O)C4CC2C3C4)=O)c2cccnc21 c1(C(=O)OC)ccc(CCC(=O)NC(C)CNC(=O)CC2CCC3CC3C2)cc1 C1(NC(CC(C)OC)=O)CCC2(CC1)CN(C(=O)CN(C)CCO)CCO2 CC1(C(=O)NC2CC(NC(C3(c4ccc(O)cc4)CC3)=O)C2)CCOCC1 C1(N(C(=O)C(C)=C(C)C)CC)CCCN(C(=O)C(C)NC(=O)NC)C1 CC1(C)CC(C)(CNC(c2ccc(Cl)[nH]2)=O)CN1C(c1cccc(C(N)=O)c1)=O C1(NC(=O)Cc2ccccc2)CCC2CN(C(=O)CSc3ccccc3)CC12 C(=O)(C(C(C)C)OC(C)=O)N1CCC(NC(C(COC(C)(C)C)OC)=O)C1 c1(C(N(C)CCN(C)C(c2snc3ccccc23)=O)=O)cc(Cl)cc2c1CCC2 C1(C(C)=O)CC(CC(N2CCCC2(C)CNC(=O)CSc2nccn2C)=O)C1(C)C c1(C(=O)NCC(C2CC2)NC(c2cc(CC)no2)=O)c[nH]c2c(C#N)cccc12 C1(C2CCN(C(c3cc(Cl)cn3C)=O)CC2)(NC(C(C)NC(CC)=O)=O)CC1 c1(C(=O)NC(C(CC)C)C(=O)NCCCC2C=NNC2=O)cc2cccnc2[nH]1 C1(N(C(C(C)CC2CC2)=O)C)CN(C(=O)C(c2ccccc2)=O)CC1O C(C(C)(C)C(C)(C)C)NC(C(Cn1cncn1)NC(COCCOCC#C)=O)=O C(=O)(CCCCCN(C(=O)C1=C(C)CC1)C)N(C1CCNC1=O)CC C(=O)(C#CC1(C)CCCO1)NCC(CN(C)C(c1ccc(Cl)cn1)=O)O Cc1ccc(C(=O)NC2CCC(C)(CNC(c3onc(C)c3C)=O)C2)nc1C N1(C(c2cccc(CC)c2)=O)CCC(C(=O)NCCOCC(C)C)=C(F)C1 c1(C(N2CCC(CCC(=O)NCCOCCF)C2)=O)ccnc(O)c1 N1(CCS(N)(=O)=O)CCCC(CNC(=O)NCCc2nncs2)C1 c1(OC)ccc(C(C(=O)NCC2CC2)N(C2CC(C)(C)C2)C)nc1C CC(C)(C#N)CC(=O)NCCC1CN(C(=O)C=Cc2cccc(CO)c2)CCO1 C1(C(C)C)CN(C(c2c[nH]c3ccccc23)=O)CCCN1C(=O)C=CCN(C)C Oc1cc(NC(c2cccc(C3CCC3)n2)c2nnnn2C2COC2)cc(Br)c1 C1(NC(C=C2CCC(C)CC2)=O)CS(=O)(=O)CC1NC(=O)C=CCN1CCCC1 c1(C(N2CCCC(NC(C(Br)=C(C)C)=O)C2C)=O)ccc2c(c1O)CCC2 C1(NC(c2c(C(C)C)cco2)=O)CC(F)CN(C(C2CC3CCC2CC3)=O)C1 c1(C(=O)NCC(CO)NC(C2CC(C)(O)C2)=O)cc(C#N)cc2ccccc12 S(=O)(=O)(c1ccc2scnc2c1)OS(CC1C(C)(C)OCCO1)(=O)=O C#Cc1cc(C(=O)NCCN(C(=O)COCC2CCCOC2)C2CC2)ccc1C c1(OCCN(C)CCO)ccc(S(N)(=O)=O)cc1.CN1CCN2C(C1)CNC2=O C1(CC)(NC(=O)Cc2cccc(C)c2C)CCN(C(C2COC(=O)C2)=O)CC1 N1(S(CC2(C(=O)OCC)CCCC2)(=O)=O)CC(C)CCC1C C(C(C(C)C(C)C)NC(C1CC(n2cnnc2)C1)=O)NC(c1n(C=C)nnc1)=O Cc1ccc(S(=O)(=O)N2CCN(C3COCC3O)CC2)c(Cl)c1 C1(NC(CCCN(C(=O)OCC)C)=O)CCCN(C(c2n[nH]c(C)c2F)=O)CC1 c1(C(=O)NCC(CNC(C(C)(C(C)C)NC(C)=O)=O)C)cnn2c(N)ccnc12 C1(C(=O)NCCC(=O)NC2CC2)CC2CCCC2N1C(C1CCC(F)C1)=O c1(C(=O)NC(C2CCCCC2)CNC(CCC(CC)C)=O)cc(C)c(C)nc1C c1(C(C)(C)NC(c2[nH]cc(OCC)c2)=O)cc(O)ccc1C(F)(F)F.NCC c1(C(N(C2CCN(C(=O)CSC)C2)CCC)=O)ccc(OC)c(Br)c1 C1(NC(c2ccc(OC(F)F)cc2)=O)CCCN(C(C2CCCC2(F)F)=O)CC1 N1(C(C(C)CC2CCCC2)=O)C2CCC1CC(NC(=O)CCc1cncnc1)C2 c1(C(=O)OC(C(=O)NCC)C)cccc2c1CCCC2 N1(C(C(C)OCCOCC)=O)CC2CC1CCN2C(c1cnc2cc[nH]c2c1)=O CC1CN(C(C2COCCN2C)=O)CCN1C(=O)CCCc1ccc(F)c(F)c1 C#CC1(C(=O)NCC(O)C(C)(C)C)CCN(C(c2conc2CC)=O)C1 N1(C(C2CNC(=O)O2)=O)CCN(C(C2(Cl)CC2)=O)CC1CO C1(C(=O)NC2(C)CN(C(c3cc(Cl)c(F)cc3N)=O)C2)CC2CCCCN2C1 CCC(C(=O)NCC(O)CNC(=O)CN(C)CC)NC(C)=O N1(c2cc(N3CCCC(CN(C)CC)C3)nc(C)n2)CCC2(CCCOC2)CC1 c1(C(N2CCC(NC(CN(C(=O)OC)C)=O)C2)=O)scc(OC)c1OC CC(C)C(O)C(C)C(=O)NCC1(O)CCN(C(=O)C=Cc2ccc[nH]2)CC1 N1(CCC)CCC(c2nnnn2C(C)C(=O)OC)(NCC2CC(=O)N(C)C2)CC1 N12CCC3C(C3C1)NC(=O)C2c1cnc(-c2cccnc2)s1.C1(COCCCl)CC1 N1(C(c2c(C)ncnc2)=O)CCCCC2(CCN(C(=O)CC3CCNC3=O)C2)C1 n1(CCCC)nc(C)c(C(=O)NCC2CCCN2C(=O)C(CCO)N(C)C)c1Cl c1(C(N(C(CNC(C2(CC)CC2)=O)C)C)=O)nn(-c2cccc(Cl)c2)nc1C C1(C(N2CC(CC(C)NC(C3CN(C4COC4)C3)=O)C2)=O)CC(C2CC2)C1 c1(N2CCC(F)(CNC(c3cc4ccsc4[nH]3)=O)CC2)nc(Cl)ncc1[N+](=O)[O-] C1(C)(NC(N(CCOCCOCC)C)=O)CCCC1O CC(CC(=O)NC1(CNC(=O)CCC(=O)N(C)C)CCC1)P(C)(C)=O c1(CC(=O)NCC(CO)NC(c2cc(C)ncc2)=O)ccc2cnccc2c1 c1(CCC(=O)NC2C(NC(CNC(CC)=O)=O)C2)ccccc1OC C1(C)(C(=O)NC2CCN(CCC)C2)CCN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CC1 CC1CCCC(C(=O)N(C2CCCC2)CCCNC(C2(CO)COC2)=O)C1 N1(C(C)C)CC(C(=O)NC(CNC(C2(C3CC3)CCC2)=O)C2CC2)CC1=O N1(C(CCCN(C(CCC(C)N(C)C)=O)C)=O)CC(O)CC(C)(C)C1 c1(CCC)c(C(=O)N(C(C)CNC(C2(NC(C)C)CC2)=O)CC)nnn1C c1(CNC(C(Cc2cc[nH]n2)NC(C(CC)O)=O)=O)ccc(C#N)s1 N1(C(C(c2cccs2)NC(C(C2CC2)SC)=O)=O)CCCC(F)C1 c1(C(=O)NCC(CNC(c2ccccc2Br)=O)OC)ccc(C#N)n1C N1(CCC(=O)NCCCNC(CCCOCCC)=O)CCCC(C(N)=O)C1 C=CCCC(C)C(C(=O)OC(C)(C)C)N1CCCC(CC(N)=O)C1 N1(C(c2cncc(C)c2)=O)CC(NC(=O)C(CO)c2ccccc2)C(C#N)C1 CC(C(=O)NCC(C1CC1)N(C(=O)CCc1ccc(F)cc1F)C)C(C)(C)C C=Cc1ccc(C(N2CCCC(NC(C3CCN(C)S3(=O)=O)=O)C2)=O)cc1 N12CC3CC1CCC3C2=O.Cn1ncc(NC(=O)COC(F)(F)F)c1C1CC1 Cc1cc(=NC(=O)C(=O)NC2CC23CCC(NC(=O)CC2CCCC2)CC3)[nH]o1 N1(C(c2cccc(C#C)c2)=O)CCC2CCN(C(=O)CC3CC34CC4)CC12 N1(C(C2CC3N(C(c4cnn(C)c4N)=O)C(CC3)C2)=O)CCc2ccc(O)cc21 c1(CC(=O)NC2CCOC(CNC(C3(F)CCCCC3)=O)C2)c[nH]c2cnccc12 Cc1ccc(F)c(Br)c1C(=O)NC1CC(NC(=O)CCC(C)(C)C)C1 Cc1ccc(C(=O)NC2(CNC(=O)C(F)(F)c3cccnc3)CCOCC2)cc1 C1(CC(=O)NCCC2CCC(NC(CSCCC(C)C)=O)C2)CC(C)(C)CCO1 n1(CC)cc(Cl)cc1C(=O)NC1(C2CCCN2C(=O)CC2C=CCC2)CC1 CN(S(N)(=O)=O)CC(N1CC(C(N)=O)(CNC(=O)CCc2nc[nH]n2)C1)=O c1(C(N(CC(CNC(C=C(C)c2ccco2)=O)C)C)=O)ccc2c(c1)OCCN2 C1(CN(C(=O)C(F)(F)C2CC2)C)CN(C(=O)COc2ccc(Cl)cc2)CCO1 C1(NC(c2c(C(N)=O)nccn2)=O)CCN(C(c2ncc(C3CC3)s2)=O)CC1O C1(C(=O)NCCC2(O)CCN(C(CC3ON=C(C)C3)=O)C2)CC2CSCC(C1)C2 Cc1sc(C(=O)NCC2CN(C(C3CC=CC3)=O)C3CC23)c(C)c1Br c1(CNC(c2nc(Cl)sc2Cl)C)c(O)ccc(F)c1F c1(C(=O)NCCCN(C(C2CS(=O)(=O)C2)=O)CC)cc(C(F)(F)F)no1 Cc1nc(N(C(=O)CCC(F)(F)F)C2C3CNCC23)nc2ccccc12 C(CC(C(=O)NCC(C1CCCC1)NC(c1ncc(C(F)F)cn1)=O)OC)OC N1(C(C(C)CO)=O)C2CCCC1CN(C(C13CCCN1S(=O)(=O)CC3)=O)C2 N1(C(c2nn(CC)c(C)c2)=O)CC(N=c2nc(S(C)(=O)=O)cc[nH]2)CC(C)(C)C1 C1(NC(C(C)COc2ccccc2)=O)CCCN(C(C2(O)CC(C)(C)C2)=O)C1 c1(C(CN(C)C)NC(=O)NCCC2CCOC2)ccc(OC(F)F)cc1 c1(C2CCN(C(c3c(C)ccnc3)=O)CC2)nc2ccccc2[nH]1 Cc1ccc(F)cc1CC(N1CCC(NC(c2cnc(O)c(C)c2)=O)C(O)C1)=O Cc1cc(C(N2CCC(C)C(NC(=O)COc3ccon3)C2)=O)cc(O)c1 N1(C(CN(C)C)=O)CCC(C#N)(NC(=O)Cc2cc(F)ccc2F)C1 c1(C(N(C2CCCN(C(C3C(C)C3C)=O)C2)CC)=O)ccc(F)c(C)c1Cl Cc1nsc(C(=O)N(CCCCNC(c2sccc2F)=O)C)c1N C1(CNC(C=COCC)=O)CCC2CN(C(C3CC4C=CC3O4)=O)CC12 c1(C(N2CCC(CNC(C(C3CCCCC3)C)=O)C2)=O)cc2cc(Cl)ccc2s1 C1(C)(NC(C2(NC(c3ccc(NC)cc3)=O)CC2)=O)CCC(C)=C(C)C1 C1(NC(c2ccccc2SCCO)=O)CN(C(=O)CC=C(Cl)Cl)C2(CCC2)C1 [N-]=[N+]=NCCCCS(=O)(=O)N1CCC(N2CCOCC2=O)CC1 N1(C(CCCCCN(C(=O)CN=c2cc[nH]cc2)C)=O)CC2CCCCCCC12 C(CC)(CCC(C)C)(c1nnnn1CCC1CC1)NC(C=C)COC Cc1cc(F)ccc1C(O)C(=O)NCCN(C(C1CC1C1(C)COC1)=O)C1CC1 N1(C(c2c(CC)ncs2)=O)CC2CN(C(=O)Cc3cc(OC)no3)CCC12 C(CC(C)(C)NC(C1CC1C(C)(C)O)=O)NC(CN(C1CCSC1)C)=O C12(C(=O)OCC)CCCC1(CNC1CCC1CO)C2 C1(CNC(C2CC(OC)C2)=O)CCN(C(=O)C(C)C2CCCC2)C1(C)C c1(C(=O)NCC(CNC(COc2cccc(CC)c2)=O)(C)O)cc(C)cc(O)c1 C=CCC(CC=C)C(=O)N(C(C)CNC(=O)C=C1CCC1)C N1(C(CC2(C)CC2)=O)CCC(C)(NC(c2cc(Cn3cccn3)on2)=O)C1 C=CCC(CC(=O)NC(C)(CO)C(F)(F)F)NC(=O)CCOCC1CCC1 S(=O)(=O)(c1ccc(Br)cc1NCC1CCC2(CC2)C1)N1CCC(=C)CC1 CCC(CCOC)C(=O)N1CCC(C(=O)NCC2(O)CSC2)C1 c1(C(N2C(C)CCN(C(CC(CCC)C)=O)CC2)=O)c(O)nnc2c1CCC2 C1(OCC(=O)N(C(C)C)CCN(C)C(C2CCC2CF)=O)CCCCC1 c1(C(=O)NCC2N(C(Cc3n(C)ncc3)=O)CC2)ccc(C#N)c(F)c1 N1(C(CNC(CC(C)C)=O)=O)CCOCC(NC(c2ccsn2)=O)C1 C1(NC(C(COC)O)=O)CC2CCC(C1)N2C(C1(OC)CCSCC1)=O CS(=O)CCC(=O)NCCC1CCCN(C(c2ccccc2OC2CCC2)=O)C1 C(=O)(C#CC1(C)CCCO1)NCC1(C)N(C(c2n(CC#C)ccc2)=O)CCC1 C(=O)(C(CO)C(F)(F)F)NCCSCC(=O)NC(C)CC(C)(C)C C(CCN=C(NCC1CCC=CCCC1)N1CCC(C(C)(C)C)C1)OCC c1(C(C(=O)NC2CCCC(NC(C(C)(F)F)=O)C2)O)cc(F)cc(F)c1 C=CCCC(C(=O)NCc1cc(C)n(C)n1)NC(C1CCN(C)C(=O)C1)=O N1(C(CC2C(CC)C2)=O)CC(NC(c2cnn(CC)c2C2CC2)=O)CC(O)C1 C1(NC(=O)Cc2c[nH]nc2O)C2CC3CN(C(=O)Cc4cccc(Cl)c4)C1C3C2 n1(CCC)ccnc1C(C1CCOCC1)NCCn1cc(Br)cn1 C12(C(N3C(CNC(CC4CC(OC)C4)=O)CCC3)=O)C(=O)C3CC1C2C3 C(=O)(C(C(=O)NCN=c1[nH]nc(CCOC(C)(C)C)s1)c1ccccc1)OCC CCC(CCCC(=O)NCCCCCN(C)CC)NC(=O)CCc1ccccn1 C1(C(=O)Nc2ccc(CC)cc2)CCC2CCC1N2C(c1ccc(CO)o1)=O C(=O)(C(CC(F)F)N(C(=O)CCC1CC1(F)F)C)NCCCCOC(C)C c1(C(=O)NCC(CO)NC(CS(=O)(=O)NC)=O)cccc2ccccc12 C(c1ccc2c(c1)CCO2)=CC(N1CC(C)C(NC(=O)CC2(C)CC2(F)Cl)C1)=O c1(OC)ccc(CC2(C(=O)NC(C)CF)CN(C(=O)Cc3ccc(F)cc3)C2)cc1 N1(C(CCC2CCC(NC(CCCOCC)=O)C2)=O)CCCNC(=O)C1CC c1(C(=O)NC2(CNC(COCC#C)=O)CCOC2)cc2c(cnn2C)nc1O N1(C(CN(C(=O)Cc2cnnn2C)C(C)C)=O)CCCCC1C c1(C(C)C)cc(N2CC3C(NC(C4(C(F)(F)F)CCCC4)=O)C3C2)ncn1 C(=O)(C1=CCCC(C)(C)C1)N1C(CNC(CC(C)n2ccnc2)=O)C=CC1 Cc1nc(CNC(c2c[nH]c(=S)cn2)=O)oc1C(=O)NC(c1cnn[nH]1)(C)C C1(N(C(C(CC2CCC2)NC(c2c(CC)ocn2)=O)=O)CC)CCS(=O)(=O)C1 C=CC(CC)CC(=O)NC(Cc1cnc[nH]1)C(=O)NCCC(=O)NCC(C)C N1(C(C(C)NC(CC)=O)=O)CCCC(NC(c2cocn2)=O)C1CC Cc1ccc(O)cc1CC(N1CCC(N(C(=O)Cc2ccccc2CO)C)C1)=O Cc1cc(C=CC(=O)N(C2CN(C(=O)C(C)N(C)C)CC2O)C)ccc1Br Cc1cc(NC(C2(C(F)(F)F)CC3CC3C2)=O)ccc1NC(=O)C(=O)NC(C)C N1(C(CC=CC=C)=O)CC2CC(NC(=O)CCSCCCC)C2C1 N1(C(CCCC2(NC(CCCCCSC)=O)CCC2)=O)CC(=O)N2CCCC2C1 Cc1nc(CO)oc1C(=O)NCC(O)CNC(=O)Cc1csc(S)n1 C(=O)(C(C)C(F)(F)C(F)F)NCCC1CCN(C(C(C(C)O)N(C)C)=O)C1 C1(CC)(CC)CN(c2nc(N(C)Cc3cnc(C)cn3)cc(C)n2)CCS1 C1(C(N(C(C)C(N2CCOC(CF)C2)=O)CCC)=O)CCN(C)CC1 c1(C(=O)NCC2N(C(CCOC(C)=O)=O)CC2)cc2sc3ccccc3c2s1 N1(C(C(C=C)CC)=O)CCCCCC(NC(=O)C(C)C2CCCC2)C1 CC(F)(F)C(C)(C)CC(=O)NC1CCC1CNC(c1cnn2ccccc12)=O N1(C(C2C3CC(NC(c4cccc(C)c4)=O)CC32)=O)CCC2(CCCO2)CC1 CC1CC(F)(F)CCN1C(C1N(C(c2cscc2Cl)=O)CC12CCCC2)=O CCCC(CCCNC(c1ccon1)=O)NC(=O)C(C(C)(C)C)c1ccccc1 C1(C)(CNC(C2(C)CNC(=O)C2)=O)COCCN(C(=O)CSCc2cscn2)C1 CC1(NC(C2CC3(CCO2)CC3)=O)CCCN(C(C2CCSCC2)=O)C1 Cc1cccc(C)c1OCC(=O)NCC1(CNC(C2CC23CC(O)C3)=O)CCC1 N1(C(c2nn(C)c(Cl)c2)=O)CCC2CN(C(=O)C(F)C3CCCC3)C2C1 N1(CC)CC(NC(c2occc2CNC(=O)Cc2coc(C)n2)=O)CCC1=O c1(C(N(CC(CC)NC(C2CC(n3cccn3)C2)=O)CC)=O)cc(Cl)cn1C C(=O)(C1=C(Cl)CCOC1)N1CCC(O)(C(CNC(c2c(C)csn2)=O)C)C1 C1(C(=O)OCC)CCC2(CNc3oc(COC)nc3C)CC12 CC1(C)CC(NC(=O)CCc2nncs2)CCN(C(c2cncc(O)c2Cl)=O)C1 N(S(=O)(=O)N(C)C)C(CNCCCC1(C(=O)OCC)CC1)C c1(N2C(c3ncc(CC)o3)CCC2)cc(-c2cccnc2)nn1C Cc1ccc(CC(N2CCC(C)C2c2cn(Cc3cnns3)nn2)=O)nc1F N1(C(Cc2c(C)cccc2)=O)CC2CCC(C1)C2C(N1C2CCC1CC(O)C2)=O c1(OCC=C)cccnc1[N+](C1(C)CCN(C(=O)OC(C)(C)C)C1)(C(=O)C1CC1)[O-] Cc1cc(C(=O)NC2CCN(C(=O)C=CCBr)C2)c(C)[nH]1 N1(C(C=COCC)=O)C2CCC1C(CNC(c1ccc(=N)[nH]c1)=O)C2 CC(C1CCCCC1)=CC(=O)NC1COC2(CNC(=O)Cn3cccn3)CC1C2 C(C(=O)Nc1cc(C)ccc1CC)(C(C)CC)NC(CC=CC=C)=O C(=O)(C(C)(C)C(C)(C)O)NCC1CC(CNC(c2cccc(C(C)C)c2)=O)C1 c1(NC(c2n(CC)ncn2)C)nccc(=NC(COC)c2cccc(Cl)c2)[nH]1 C1(NC(c2c(CC=C)cccc2)=O)CCN(CC(=O)NCC2CC2)C(C)C1 C1(C(=O)NC(C2CCCN2C(c2ccc(SC(F)(F)F)o2)=O)(C)C)CCCCS1 C1(C(=O)OC)CC(C)N1C(=O)C(CC1CC1)NC(=O)CCOCC(C)(C)C c1(C(=O)OCC(C)CO)cc2c(s1)CCC(C(C)(C)C)C2 C1(C(=O)NC2CC(Cn3cc(C4CC(F)(F)C4)nn3)C2)CC12CCOC2 c1(C(C)=O)nccc(SCC(O)CO)c1F CC(F)(F)CCC(=O)NC1CC2CC1N(C(C1CCCC1(C)C)=O)C2 C1(CC(N2C(C(N(CCCC)CC)=O)CSC2)=O)CC=CCN1C N1(C(c2cc(C)on2)=O)CCCOC(CNC(=O)CC(C(F)F)c2ccccc2)C1 CCC(C(=O)N1CCC(NC(C2(C(F)F)CCCCC2)=O)C1)C(F)(F)F C(=O)(C(C)(C)CS(C)(=O)=O)N1CCC(F)(CNC(CCC(CC)C)=O)C1 C(=O)(C(C)(C)C(=O)N(C)C)NCc1ccc(C(=O)NCC(CC#C)(C)C)o1 CC(CN=c1[nH]cnc2c1CCCC2)NC(=O)COc1cnn(C)c1 C(C1CN(C(c2ccncc2O)=O)CC1C(=O)N(c1ccccc1)C)=CC N1(C(C=CCC)=O)CCCC(C)(CNC(c2c(OC)ncnc2C)=O)C1 c1(OC)c(C(=O)NCC2CN(C(C3OCCO3)=O)CCO2)c(C)nn1C CC#CCCCC(=O)NC(CCC1CCC1)C(=O)NCc1ccc(OC)cn1 CC1CCC(C)CN1C(=O)CCNC(c1ccncc1N)=O N1(C(c2cncc(OC)c2C)=O)CCC(C)N(C(C2C=CCCC2)=O)CC1 c1(NC(C(=O)Nc2c(CC(=O)OCC)scc2)=O)cn(CC2CC2)nc1C c1(C(=O)NC2CN(C(C(CCC)OCC)=O)CC2O)ccc2nnnn2c1 C1(C(=O)NC2CCCN(C(C3CCC(O)C3)=O)C2)CCn2nnnc2C1 C1(NC(=O)C=CCBr)CN(c2ccnc(C3CC3)n2)CC1F Cc1cccc(OCCC(=O)N2CC(CCNC(=O)CCNS(C)(=O)=O)C2)c1C CCC(C(=O)N1CCCC(COC)(NC(c2cncc(OC)c2)=O)C1)C(C)C C1(CNC(C(CC)C)=O)CCN(C(=O)CCC(C)C)CC1O C(=O)(CS(=O)(=O)CC(C)C)NC(CCOC)CNC(C1(C)CCN(C)C1)=O C(C)(C)(CN=c1[nH]c2ccc(OC)cc2s1)NC(COCCOC)=O Cc1nc(C(=O)NC2CC(NC(c3cc(CC4CCC4)c[nH]3)=O)C2)cn1C(F)F C12(C(=O)NCCC(C)(C)NC(CC(C)F)=O)CCC(N(C)C)(CC1)CC2 N1(C(CCSCCCC)=O)CC(NC(=O)CC(C)C(C)C)C(C)(C)C1 c1(C(=O)NC2CN(C(C3CCc4n[nH]cc4C3)=O)C2)c(F)ccc2nc[nH]c12 C1(C(N2CC(C#C)(F)C2)=O)CN(C(=O)CCC(CC)CC)CC1N=[N+]=[N-] CON(C)C(=O)C(CC(C)C)NC(c1cnccc1C#N)=O C12(CNC(C(C)C3CCC3)=O)CCC(CC1)N2C(C1(C(=O)OC(C)(C)C)CC1)=O C1(O)(CC(=O)NCC2C(C)(C)C2C(=O)NCc2nccs2)CCCOC1 c1(CC)cc(CC(=O)NC(C)(CNC(=O)CC(C)C=C)CO)n(C)n1 C1(OC)(CNC(C2SCCCS2)=O)CCN(C(c2ccncc2)=O)C1 c1(C(=O)NCC2(C)N(C(CCOC)=O)CC(F)(F)C2)ccc2c(c1)CCCS2 c1(COC)ncc(C(=O)NCC2CCN2C(=O)CNC(=O)CC(C)C)cn1 c1(C(N)=O)cccc(C(=O)NCC(F)CNC(C2CN(C3CCC3)C2)=O)c1 C(=O)(CC(C)(C)CCC)NC(CC#C)(C)C(=O)NC1CC1c1cnn(C)c1 C(CNC(C(C)(C)OC(C)=O)=O)(C(C)C(C)C)NC(=O)NC(=O)C=C(C)C(C)(C)C CC(C(=O)N(C1CCCC1)CCNC(c1ncccc1F)=O)C(C)C(C)(C)C CC1=NNC(=O)C1CCC(=O)NCC1(C)CC(NC(C2(O)CCCCC2)=O)C1 C#CC1(NC(=O)C(c2ccco2)NC(=O)C2=CCCOC2)CCCOC1 C1(c2nnnn2-c2ccc(F)cc2)(NCCOCCCC)CSC2CCCC12 N1(C(C23CCC(CN(C(CC4CC(CC)C4)=O)C2)C3)=O)CCc2nn(C)cc2C1 c1(CCC)ccccc1C(=O)NC(Cn1cncn1)C(=O)N1CCC1CC1CC1 N1(C(C2CC3CC3N2Cc2c(F)cccc2Cl)=O)Cc2ccc([N+](=O)[O-])cc2C1 c1(C(=O)NC2CCN(C(=O)OC(C)(C)C)CC2)ccc2cccnc2c1F N1(C(C2(C#N)CCCC2)=O)CCC2(CC1)CC2NC(c1cccc2ncsc12)=O CCCC(C)CC(=O)NC1CCC1CNC(=O)CNC(c1cnoc1C)=O c1(C(N2CCC3(NC(c4ccc(Cl)cc4Cl)=O)C(C2)C3)=O)ccnc2[nH]cnc12 CC(C)(CCCC(=O)NCC1(CO)CC=CC1)NC(=O)Cc1cc[nH]n1 c1(OC)ccc(C(=O)NCC2CC(F)CN2C(c2cncc(CO)c2)=O)cc1O c1(N2C3C(N4CCN(CC4)C(OC)C2)C3)cccc([N+](=O)[O-])c1.OC N1(C(CC2(C=C)CCCCC2)=O)CCN(C(C2CC(=O)N(OC)C2)=O)CC(C)C1 C1(NC(c2c(C)nc[nH]2)=O)CCCN(C(=O)C(C(C)C)N(C)C)C1C Cc1ccc2nc(SCCC(=O)NCCC3CC(NC(C4CC4C)=O)C3)[nH]c2c1 C1(C(=O)NCCN(C)C(C2CCN(C)S2(=O)=O)=O)CCS(=O)(=O)C12CCC2 Cc1cc(CNC(c2ncncc2-c2cccc(F)c2C)=O)cnc1C N1(C(C2(CC)CN(C(=O)Cc3cccnc3O)C2)=O)CCN(C)C(=O)C1C N1(C(=O)CC2COCCO2)CC2CN(C(c3cccc(C(N)=O)c3F)=O)CC2C1 C(=O)(CCC1=NNC(=O)CC1)NC(CC1C(C)(C)C1)=O.C12CCN1C2 C1(NC(c2cc(C(C)(C)C)on2)=O)CCN(c2ncncc2Cl)CCC1CO CCC(C)C(C(=O)N1CCC(=CCNC(=O)Cc2cc(C)ccc2F)CC1)OC C1(NC(c2cc(C)[nH]c2)=O)CCCC12CCN(C(c1conc1C(C)C)=O)CC2 c1(C(N(CCCNC(c2cnn(C)c2C)=O)CC)=O)c(C)nn2cc(C)cnc12 c1(C(=O)NCC2CCSCC2)c(-c2cnc(F)c(F)c2)cncc1F c1(CC(=O)NC(C)(CNC(=O)C(F)CN(C)C)C2CC2)ccc(F)c(Cl)c1 C1(C(=O)NC2(CO)CN(C(C(Br)=C(C)C)=O)C2)Cc2ccccc2N1C C1(N(CC#C)C(c2cc(Cl)cs2)=O)CCN(C(C2CCS(=O)CC2)=O)CC1 C=CCC(CC)C(=O)Nc1cccc(C)c1.C1(=O)C(NC(=O)OCCOC)CN1 N1(C(c2cccc(C(C)C)n2)=O)CCCC(N=c2nc(C3CC3)[nH]s2)C1 N1(C(=O)Cc2cccc(F)c2)CCC(O)C(CO)C1 Cn1cc(S(N)(=O)=O)cc1C(=O)NCCCNC(=O)CC(F)(F)c1ccccc1 c1(CC(=O)NC(CC)(C)CNC(c2csc(Cl)c2)=O)ccc(-n2cccc2)cc1 C1(NC(C2N(C)CCC2)=O)CCN(C(C2OCC3CCCC2C3)=O)CCC1(F)F C1(C(=O)NC(C2CCCC2)CNC(=O)C=CC(C)(C)SC)(OC)CCCCCC1 C1(C(=O)NC(COC)C(C)C)C2CC3C(C2NC(=O)CSc2nc[nH]n2)C13 c1(C(N2CCN(C(C3C(C(N)=O)C3)=O)CC2CC2CC2)=O)ccnc2[nH]cnc12 c1(C(N2CCC(CN(C(C3C(C=C)CC3)=O)C)C2)=O)cc(O)nc2c1CCCC2 C1(C(=O)NC)CCN(c2cc(NCC3CC34CCC4)ncn2)CC1 C1(NC(CCN(C(CC)CC)C)=O)CC2CC(NC(=O)CSCCN(C)C)CC12 O=C(C(CC(F)(F)F)c1ccc(F)cc1)Nc1cc(F)c(Cl)cc1Cl N1(C(c2cnc(C)n2C)=O)CC2CCCC(N(C(=O)COc3ccsn3)C)C2C1 c1(-c2cc(C(=O)NCc3n(CCC)ccn3)n[nH]2)c(C)nn(C)c1C c1(C(N(CC(C)NC(C2CCOC2c2ccccc2)=O)C)=O)cc(N)cc(F)c1 N1(C(c2c(C)oc(Cl)n2)=O)CC(C2CN(C(=O)C=Cc3ccc(C#N)cc3)C2)C1 C1(NC(C2(F)CN(C(c3cnn(C4CC4)c3)=O)C2)=O)CCCC2(C1)N=N2 C#CC1CCCN1C(c1scc(-c2ccc(F)cc2)c1C(=O)OC)=O c1(C(N2CC3C(C(N(CC)CC)=O)(C3)C2)=O)ccc(OC)c(F)c1F c1(CCC(=O)NC(CNC(CCC#CC)=O)C)ccc(F)c(OC)c1 c1(OC)cccc(C(N2CCN(C(C)C)C(C(=O)OC)C2)C(=O)O)c1Br C(=O)(C(C)(F)C(=O)NCCN(C(=O)C(C)OCC1CC1)CC1CC1)OC Cc1occ(C(=O)O)c1CN1CCCC1c1ccccc1C(F)(F)F C1(NC(CCNC(C)=O)=O)CC(NC(c2sc(N(C)C)nc2C)=O)C12CCC2 N1(CC)CC(C(=O)N2CC(O)(CNC(=O)CC3=CCCCC3)C2)c2ccccc21 CCC(C)(CC)C(=O)N1CC(NC(=O)CC2SC(=N)NC2=O)C(n2cccn2)C1 C1(NC(C2C(=C)CC2)=O)CCN(C(=O)CSCCC#N)C(C)C1 CCC1=C(C(=O)NCCN(C(c2c(F)cccc2Br)=O)CC)CCCO1 N1(C(C(CC)C)=O)CC2(CCNC(=O)C3=CCCS3)CCC1CC2 C(=O)(C1=CS(=O)(=O)CCC1)N(CC(C)O)CCNC(=O)C=CC1CCCC1 C12(C(=O)Nc3ccc(C)cc3)CCC(CC1)N(C(C13CC1CNC3=O)=O)C2 Cc1ccc(NC(=O)CC2CCN(C(=O)Cc3ccc(F)c(C)c3)CC2)c(Br)c1 C(=O)(C1=CS(=O)CCC1)NC(C(C)C)CCNC(c1ncccc1C(C)(C)C)=O C(C(C)S(N)(=O)=O)NC(CCN(C(=O)CCOCCCOC)CC=C)=O N1(C(c2c(C)[nH]cc2)=O)CCC(CNC(=O)C(C)OCC2CC2)C(C2CC2)C1 C1(NC(Cn2nc(C)c(Cl)c2)=O)CC(CNC(=O)CN(C)C2CC2)C12CCC2 Cc1noc(C)c1C=CC(=O)NCC1CCCC1NC(=O)Cc1nc(=N)[nH][nH]1 N1(C(C#CC(C)C)=O)CC2CC1CN(C(c1cccc(F)c1Br)=O)C2 C(C)(C)(CC(=O)N1CC(F)CC1CNC(=O)CCCc1csc(=N)[nH]1)SC N1(C(C(C(C)C)C)=O)CCN(C(=O)Cc2ccccc2CC#N)CC1CCN(C)C C1(NC(=O)CCc2ccccc2)CC12CCN(C(=O)CC1CCSCC1)C2 c1(C(N2CC(NC(C(C(C)C)SC)=O)C2)=O)cc(O)c2c(cnn2C)c1 c1(C(N2CCC(CCC(=O)NCCC(CCC)C)CC2)=O)ccc(C)c(F)c1 c1(C(=O)NC)ccc(C=CC(=O)NC2CCCC2NC(C2CCC2C)=O)cc1 N1(C(c2[nH]cc(C(N)=O)c2)=O)CCCN(C(=O)C=CSc2nc[nH]n2)CC1CO C1(c2n(C)ncc2)CN(C(=O)CCc2ccc[nH]2)CCN1C(=O)C1CC1 N1(C(c2c(C(C)C)c(F)ccc2)=O)CC(C2CN(C(=O)COC3CCCC3)C2)C1 c1(C(N2C(CC)CN(C(=O)CC3CCC3)CC2)=O)cc2c(nn1)OCCS2 C1(F)(C(N2CCC(CNC(=O)CC3CCNC3=O)C2)=O)CCS(=O)(=O)C1 C1(C(N2CC(NC(c3n(C)ncc3)=O)CC(C)(C)C2)=O)CC2CCC1CC2(F)F c1(CCCC(=O)NC2CC(n3cc(CCOC)nn3)C2)ccc(Br)cn1 c1(CC)n[nH]cc1C(=O)NCCCCNC(c1n[nH]cc1Cl)=O N1(C(CNC(COCCSC)=O)=O)CCN(C(C2COCCC2C)=O)CC1 C12(NC(C(=O)NCC)=O)CCCN(C(c3nc(O)sc3C)=O)CC1C2 N1(C(c2cc(OC)no2)=O)CCCN(C(C2CCCO2)=O)CC1CO N1(C(=O)NCCCCCCCC)CC2(CCCN2C(c2nccnc2OC)=O)C1 C1(CC)C(NC(C2CCCN2C2CCCCC2)=O)CCN1C(=O)Cn1cncn1 C1(C(=O)Nc2cncc(C(N)=O)c2)CC12CCN(C(c1ccc(F)c(O)c1)=O)C2 C12(CNC(C(C)(C)NC(=O)NCC)=O)CC1CN(C(=O)Cn1cccnc1=O)C2 Cc1cnncc1C(=O)NCc1ccnc(C(=O)NC(c2nnc(O)n2C)C)c1 c1(C(=O)NCCCC(C)(C)NC(c2c(C)nc(C)[nH]2)=O)ccc2sc(O)nc2c1 N1(C(C2CC23CCOCC3)=O)CC2(CCCCN2C(=O)CCF)C1 c1(C(N2CCN(C(c3c(C(C)C)ccs3)=O)CC2)=O)cc(Cl)cc(C(F)(F)F)n1 c1(C(c2ccccc2)N(C(=O)CC2CCC(C)O2)CC)ccccc1C C(=O)(C(CC(C)(C)C)NC(=O)Cc1ccoc1)NC(CC(C)C)CO C1(C)(C(N(CCCNC(=O)CC2CCC3CC23)CC)=O)CCC(=O)C1 CC1CN(C(=O)CCCC(N)=O)CCC1CNC(=O)C=C1CCCCC1 N1(C(COCCC=C)=O)C2CCC1CN(C(C1CCN(CCO)C(=O)C1)=O)CC2 C1(C(N(CCCN(C(C2C(C)=C2)=O)C)C)=O)(NC(N)=O)CCC1 c1(N2CCN(C(C)=O)CC2)nc(N2CCOC(c3cn[nH]c3)C2)nc2scnc12 c1(C(C2CCOC2C)N(CC(F)(F)F)CC)ccc(Cl)cc1 N1(C(Cc2cc(C)on2)=O)CCC2(NC(=O)Cc3ccccc3C(C)C)CC2C1 c1(SCC)ccc(CC(=O)NC)cc1.C1CCCCN1C(=O)CC1(CC)CCC1 C1(CC(=O)N(CCCNC(=O)CC2CCC(=O)N2C)CCC)CC2(CCC2)CO1 CC1CCC(NC(c2ccc(OCF)cc2)=O)CN1C(=O)CC1CC2(CC2)C1 C=C1CC2(C1)CC(C(=O)N(CCN(C(=O)CCC(C)SC)C)C(C)C)C2 N1(C(C(c2ccccc2)C)=O)CC(CNC(=O)CCC2CC(F)(F)C2)C2(CC2)C1 CC(C)C(=O)C(=O)NC(C1(C(=O)N(C2CCCC(O)C2)C)CC1)C c1(OC)cc(CN2CCN(C(=O)C(=O)NCc3ccccc3F)CC2)ccc1C C(=O)(C(C#N)C(C)C)NCC1N(C(CCC=C)=O)CCOC1 C1(NC(=NC)NCC2CC(F)(F)C2)CCN(CC)CC1C CCCCCCCCC(F)C(=O)NCC(O)CCNC(c1c(C)nsc1N)=O c1(CNC(CC)(CSC)c2nnnn2C2CCC2)noc2c1COCC2 CC(CSc1ccccc1)C(=O)NC(CNC(=O)COCC(C)(C)C)C1CCC1 c1(CNC(C2C(CC)N(C(c3cc(OC)n[nH]3)=O)CC2)=O)cnnc(C)c1C c1(OC)nccnc1C(=O)NCCC1CCCN1C(C1CC(=O)N(C)C1)=O c1(C(=O)NCCC(CNC(C(C)OC2CCOC2)=O)O)ccc2c(c1)CC(=O)N2 C1(OCC(=O)NCC2C=CCN2C(=O)C=CCCc2ccccc2)CCOCC1 Cc1cccc(S(=O)(=O)CCCN2CCCC(N(C)Cc3cnc(C)cn3)C2)c1 CCCC(CC(C)C)C(=O)N1CC(OCC(=O)NC(CC2CC2)CC)C1 C(=O)(CC(C)CNC(=O)C(=O)NC1CC2C(CO)C2C1)OCC CC1(C)OCc2cnc(NC(C3CCC4(C3)OCCO4)=O)nc21 Cc1ccc(=O)n(CC(=O)NC2CC(C)N(C(c3cccc(C4CC4)n3)=O)C2)n1 C1(SCC)CCC(F)(F)CC1.N12CCN(CC1)C(=O)C1(n3cnc(n3)C2C)CC1 c1(C(=O)NC2CC(C(C(=O)NC(c3ncc(F)cn3)C)F)C2)c(C)nn(C)c1N CCCC(C)(CCC)C(=O)NC1CC(C)(NC(=O)C=Cc2nnc(C(C)C)o2)C1 c1(C(N(C(C)CC(=O)N2CC(c3ncc[nH]3)C2)C)=O)cccc(F)c1 N1(C(c2ccccc2SC(F)F)=O)CC(NC(C2CCCOC2)=O)CC(F)C1 c1(OC)ncc(NC(C2CCN2Cc2cncs2)=O)cc1C c1(C(=O)NC(CCOC)CNC(C2CC(CCO)C2)=O)cccc(OC(F)F)c1 C(=O)(C1=NN(c2cccc(C)c2)C(=O)CC1)NC1C2CN(C(CCC)=O)C1CC2 C(=O)(CS(=O)(=O)c1ccccc1C)NC(CC)CNC(c1cc(N)ccn1)=O CC1CN(C(c2ccn(C)n2)=O)CC(C)N(C(c2ccc(Br)cc2N)=O)C1 N1(C(C(C)OC)=O)CC(C)(C)CC1CNC(C1(CNC(=O)OC(C)(C)C)CCC1)=O N1(C(Cc2cc(C)[nH]n2)=O)CCC(N(C(=O)CCc2ccccc2Cl)C)C(C)C1 CCCC(O)CC(=O)NC12COC(CNC(=O)C(C)C3CCC3)(C1)C2 Cc1cc(C)n2ncc(C(=O)NC34CCCN(C(=O)C=CCF)CC3C4)c2n1 C#CC1CN(C(=O)C(c2ccco2)NC(C2CCCC3(CC3)C2)=O)CCO1 C(=O)(C(F)(F)C1(O)CCC1)NCC(C)(C1CC1)NC(c1ccc(C(F)(F)F)s1)=O C1(C(=O)NC(C(C)NC(C(C=C)CC)=O)CO)Cc2ccccc2C1 CC1CC(NC(c2ccon2)=O)CCN1CC1CCCS(=O)(=O)C1 C1(CNC(C(=O)NCC2(CCOC)CCOC2)=O)C2CCC(CC2)C1C(F)(F)F Cc1ccc2c(c1)C=C(C(=O)NC1CC(N(C)C(C3CCCC3(F)F)=O)C1)CO2 Cc1nc(C)c(C(N2CCC(c3cc(CNC(=O)C(C)N(C)C)on3)CC2)=O)[nH]1 n1(CC)cc(C(=O)NC2CCCC2CNC(=O)CCCc2ncc(C)o2)cn1 N1(C(C(C(=C)C)(C)O)=O)CCC2(CC1)CC(C)N(C(c1cn(C(C)C)cn1)=O)C2 C12(C(=O)NCC3=CCN(C(CCOCCC)=O)CC3)CCCN(CCC1)C2 c1(NCC)cncc(C(=O)NC2CN(C(c3cn(C4CC4)nn3)=O)CC2C)c1 C1(CN(C(=O)C(O)C2CC2)CC)CCN(C(=O)CCc2cscn2)CC1 C(CC(C)(C)CC(=O)NC1CCN(C(C2CC2(F)F)=O)C(C)C1)OC c1(C(=O)NC2CCN(C(C(=O)NCCCC)C)CC2C)cccc2nn[nH]c12 N1(C(C=C(C)Cl)=O)C2CCC1CC(NC(c1n[nH]c3c1CC1CC31)=O)C2 n1(CC(=O)NCCC2CC(NC(C3CCO3)=O)C2)ccc(Br)cc1=O O=C(C1=CCCCO1)C(CCNC1C=CCC1)=O.C1(N)CC1 C1(CC=C)(NC(=O)C=CCN(C(=O)CCC=CC(C)C)C)CCOC1 C(=O)(C(F)CC(C)(C)C)NCC1(NC(c2cc(C)[nH]c2C)=O)CCCCC1C C12(CNC(C(c3n(C)ncc3)O)=O)CCCC(CN1C(=O)C=CCO)C2 c1(C(C(=O)NCc2ccc(C)cc2)N(C2CC(=O)NC2=O)CC)cccc(Br)c1Cl Cc1nn(C)c(C)c1CN(C(=O)CC1CCCCC1F)C1CC1 C(=O)(C(CCS(C)=O)N(C)C)NCC1CCC(NC(CCCNC(C)=O)=O)C1 c1(CC(=O)NC2(CC(=O)N(CCCN(C)C)C)CCC2)ccc(Cl)s1 C1(C(=O)N)(NC(CSCC#C)=O)CCN(C(=O)Cc2ncc(C)s2)C1.OC N1(C(C(COCC)n2cc(C(O)C(C)(C)C)nn2)=O)CC(C)(C)C1C(C)C c1(C(N2C3C(NC(CCN(C)CCO)=O)C(C3)C2)=O)cc2c(nc1O)CCOC2 N(C(=NCCc1ccccc1)NCC1CCO1)CC(C)N(C)C C12(NC(CCN(CCCCC)C)=O)CC(C1)N(C(C1CCCOC1)=O)C2 C1(NC(c2ccc3cccnn23)=O)CC2CC(C1)N(C(=O)C=C1CCCC1)C2 c1(CN(C(=O)NC2C(OCC)COCC2)C2CC2)ccc(Cl)c(Cl)c1 N#Cc1ccccc1C(=O)NCCN(C(C1CC1c1ccco1)=O)C1CC1 C=C=CCCC(=O)NC1(C)CCN(C(=O)C(C)(C)n2cc(Br)cn2)C1 c1(C(N2CC(N3CCN(C(c4cnn(CC)n4)=O)CC3)C2)=O)coc2c1CCCC2 C1(CNC(C2CCC(N(C)C)C2)=O)C2CN(C(c3cc(Br)n[nH]3)=O)CC12 c1(CC(=O)NCc2ccccn2)cc(Br)ccc1Cl C(CC)(CC(F)(F)F)NC(C#CCNC(C(COC)N(C)C)=O)=O C1(C(=O)NCC)(CNC(c2nnnn2C(C)(C)CC)C2CCSC2)CCCC1 C(=O)(N=c1nc[nH]n2cccc12)C1C(NC(C(CC(C)C)O)=O)CC(C(=O)O)CC1 C1(CC(=O)NC2CCCN(C(C3(C)COC3)=O)C2)CN2CCN1CC2 c1(C(N(C2CCN(C(=O)Cc3csc(Cl)c3)C2)CC)=O)cc(C)cc(C)n1 c1(CC)c(C(=O)N(C2CCN(C(=O)CCSc3nccn3C)C2)CC)ccn1C c1(NC2(C3CN(C(=O)CCC4CCC4)C3)CC2)ncnc2ccc([N+](=O)[O-])cc12 Cc1c(C(=O)NCC(C2CC2)NC(c2cnn(C)c2Cl)=O)[nH]c2cc(F)ccc12 c1(C(N2CCC(NC(=O)COCC(F)(F)F)(CO)C2)=O)cnn2cccnc12 CC1(NC(C2(c3ccccc3)CC2(F)F)=O)CCN(C(=O)CS(N)(=O)=O)CC1 Cn1ccc2cc(C(=O)NC3CC(O)CN(C(=O)CSC(F)F)C3)cnc12 CCC(O)C(F)(F)C(=O)N1CC(CCNC(c2cnn(C(C)C)c2C)=O)C(C)C1 CCCCC(C)(C)NC(=O)C(C)C(C)NC(=O)CC1CCN(C)CC1 c1(OC)cnc(C(=O)NCC2CN(C(c3cc(C)n(C4CC4)n3)=O)C2)cn1 c1(C(=O)NC(CC)CN(C)C(C2(N=[N+]=[N-])CC2)=O)cc(C)nn1C1CC1 C1(NC(c2cncc(OC)c2)=O)CN(C(C2CCOC(C)(C)C2)=O)C2(CCC2)C1 C1(C)(CNC(C(C(C)C)C)=O)CN(C(=O)CCc2cncc(O)c2)CCO1 C1(NC(=O)Cc2cnns2)CC2CCCC(C1)N2C(C1(CF)CCC1)=O C1(CCNC(C(c2cccnc2)C)=O)CCCCN1C(=O)CCc1cnc(O)[nH]1 c1(C(CNC(c2ccc(C(C)(F)F)cc2)C)=O)ccc(F)c(Cl)c1 c1(C(N2CC3(CCN3C(C3CCCC34CC4)=O)C2)=O)cccc(Br)c1F Cc1ccc(C(N2CC(NC(=O)Cc3cccnc3Cl)C3CC23)=O)c(C)n1 C1(CNC(C(CC)(C)C)=O)CCC2(CCC2)C1NC(=O)CC(F)(F)CC C1(NC(C2N(C(CC)=O)CSC2)=O)COCCC1NC(C1CCC(C)CC1)=O Cc1ccc(C(=O)NCCCNC(c2ocnc2C(F)(F)F)=O)cc1S(C)(=O)=O S(=O)(=O)(c1ccc(=NCCc2ccc(N(C)CC3CCSCC3)cc2)[nH]c1)NC CC(C(=O)NC1CCOCC1NC(c1c(Cl)nn(C)c1Cl)=O)C(C)(C)C CC1(C)OCC2CC12C(=O)NC1(CNC(c2nccc(Cl)c2O)=O)CCOC1 CC(CNC(=O)C(c1ccn(C)n1)C)CC(=O)NC(c1nc[nH]n1)CO c1(C(N2C(C(C)(C)NC(c3ccc(Cl)o3)=O)CCC2)=O)cc2ccc(F)cc2[nH]1 c1(C(C(=O)NC(CN(C(=O)C(n2nccc2C)C)CC)C)(C)C)ccc(Cl)nc1 Cc1cccc(C(N2C3CCC2CN(C(C2COC(=O)N2)=O)C3)=O)c1[N+](=O)[O-] N1(C(c2c(C)nc(O)[nH]2)=O)C(C)CC2CN(C(c3csc(=N)[nH]3)=O)CC12 C1(C)(COC)CC(NC(c2ncc(F)cn2)=O)CN1C(c1c[nH]nc1OC)=O CC(C(C)C(=O)NC(C)(C)C(=O)NO)NC(=O)Cc1cn(C)cn1 C1(NC(Cc2cc(=N)[nH]cc2)=O)CC12CCC(NC(c1cc(CO)[nH]n1)=O)CC2 c1(SC)ccc(C(N2CC3CN(C(=O)C(C)Cc4ccco4)C3C2)=O)cc1F CC(C)(C(=O)NCc1cc(C(=O)NCC2(F)CC(O)C2)no1)C1CCCO1 CCCC(O)C(CO)NC(C1(NC(c2nc[nH]n2)=O)CCCC1C)=O Cc1ccc(S(=O)(=O)O)cc1NC(C1C=CCN1Cc1c(O)cccc1Br)=O c1(C(=O)NC(C2N(C(C3CC(SC)C3)=O)CCC2)C)n[nH]c(C)c1Cl N1(C(CCn2c(C)nc(C)n2)=O)C2CCCC1CC(NC(=O)C(O)CC(C)C)C2 N1(C(CCCOCC=C)=O)CCOCC(NC(C2COC(C)(C)CO2)=O)C1 CC1CC(NC(c2cccc(C(N)=O)c2)=O)CN(C(=O)Cc2ccsc2)C1 C(=O)(C#CC1CCCOC1)NC(C1CCCN1C(C1OCCC1(C)C)=O)C C(CC(C)(C)C)(C(=O)NC1CCOCC1C(=O)NCCOCCN=[N+]=[N-])OC c1(C(=O)NC2(CO)CN(C(C(C(CC)(C)C)O)=O)C2)ccc(S(N)(=O)=O)cc1Cl N1(C(CCCCC=C)=O)CCC2(C1)CN(C(c1cc([N+](=O)[O-])n(C)n1)=O)C2 c1(CC(=O)NC2(CN(C)C(c3cc(F)cnc3O)=O)CC2)ccc(C#N)nc1 C(N=c1ncc(F)c[nH]1)C1C(NC(CN(C2CCC(C)(C)OC2)C)=O)CCCC1 CCCCCC(O)C(=O)N1CCCCCC1CNC(c1cc(O)nc(CC)n1)=O CN1CCOc2ccc(C(N3CC(O)(CCNC(C4CC45CCC5)=O)C3)=O)cc21 N1(C(c2cccc(OCC)c2)=O)CCN(C(C2(F)C3CCCC23)=O)CC1CO CCC(CC(=O)N1CCC(OCCNC(C2OCC2(C)C)=O)CC1)C(C)C N1(C(c2occ(C)c2C)=O)CC(NC(C2CCC(C)(C)C2)=O)C(C2CC2)C1 C1(C(=O)NC(c2ccccc2)C#C)(NC(=O)C(C)OCC2CC2)CCSC1 c1(C(N(CC(C)NC(c2c(CCC)cccc2)=O)CC)=O)c(C)cc(=O)oc1C C1(CCC)(NC(=O)CCC2CC2(F)F)CCCN(C(=O)C#CC(C)(C)O)C1 C(=O)(C(CCOCC)NC(c1ccn(C(C)C)n1)=O)N1CCC(CC)C1 c1(C(=O)NC(CCOCC)C(=O)N(C)CC2CC2(F)F)cnc2cc[nH]c2c1 C1(NC(c2scc(C(C)=O)c2)=O)CN(C(C2CC2c2ccccc2)=O)CC1OC C1(NC(=O)CC2COCCN2Cc2ccc(OC(F)F)cc2)CCCCC1(F)F C(=O)(C(C)(C)CC1CCC1)N1CCC(N(C(C(C)C)=O)C)C1 CC(C)(C)CC(=O)NCc1ccc(CNC(=O)C(O)CN2CCOCC2)cc1 N1(C(C(CCOCC)NC(C2CC(OC3CC3)C2)=O)=O)CCC12CCOCC2 CCCCCC(O)C(=O)NC1CCCCN(C(c2cscc2C(=O)OC)=O)C1 c1(C(=O)NCC(C)N(C)C(C2CCCO2)=O)cnc2ccc(Br)cc2c1 C(=O)(C(CO)C(C)(C)C)NC(C)CC1CN(C(C2COCC2(C)C)=O)C1 c1(CC)cc(C)ccc1C(N1CCC(CNC(=O)CC2CCOC2)C1)=O c1(C(=O)NC2CC(CNC(C(c3cn(C)nc3)=O)=O)C2)cc2n(c1)CCCC2 c1(C(=O)NC(CC)CNC(=O)C2=CCCC2)cc2cnn(C)c2s1 c1(C(=O)NCC(CNC(C(C(CC)C)O)=O)(C)O)ccc(Cl)c(O)c1N C1(NC(CC2(C(=O)OCC)CCC2)=O)CCCN(C(c2csc(C)c2)=O)C1 N1(C(C2CC(C)OC2)=O)C2CCC1CC(CNC(c1cc(C(F)(F)F)cs1)=O)C2 C1(OC(C2CCN(c3ccncn3)C2)=O)CCC2CC2CC1 C12(C(=O)NCC3(F)CCN(C(c4c(C(C)=O)ccs4)=O)C3)CC1COC21CCC1 N1(C(C(=O)NCC)C2CC(C(=O)OC(C)(C)C)C2)CCN(c2ccncc2)CC1C N1(C(C(CC2CC2)OC)=O)CCC(C(=O)Nc2ccsc2C(N)=O)(OC)C1 N1(C(c2ccc(CC)cc2)=O)CC(CNC(C2C3CCCC23)=O)C(F)(F)C1 c1(C(=O)NC(CC(C)NC(c2ccsc2C(F)F)=O)C)cccn2cncc12 Cc1c(Cl)sc(Cl)c1C(N1CC(F)(CNC(C2(C(C)C)CC2)=O)C1)=O c1(C(N2C(CNC(c3c(CC)n(C)cc3)=O)CC2)=O)ccc2c(c1)C(=O)CCN2 c1(C(N2CCN(C(CCCCC#C)=O)CC2CO)=O)noc2ccc(Cl)cc12 c1(OC)nc(C(=O)NCCN(C(=O)CC2CC2C)C(C)C)ncc1F C1(C(N(C)CC2N(C(C=Cc3ccc(C)o3)=O)CCC2)=O)Cc2ccncc2N1 c1(SN2CCCC(C)(c3cc(C)[nH]n3)C2)cc(F)cc2c1CCC2.C(F)(F)F C1(CCC(=O)NC(c2ccncn2)C)CCN(C(C2(C)CCCS2)=O)CC1 c1(CC(=O)NC2CC(CNC(CN(C)C(c3cccs3)=O)=O)C2)sc(O)nc1O CCCCC(CC)C(C(=O)NCC(F)F)N1CCC(C(O)CSC)CC1 c1(SCC(N2CCN(CCCN3CCCNC3=O)CC2)=O)cc(F)cc(F)c1 C1(NC(C(CC)OC)=O)CCC(CC(=O)N(CCCO)C(C)C)CC1 C=CCCC(F)(F)C(=O)NCC1(CNC(C2CC3CC2CC3O)=O)CCC1 c1(C(=O)NCC(C)N(C(=O)C(C)c2ccco2)C)ccc2ncccc2n1 c1(NC(C(=O)NCc2cccc(SC)c2)=O)ccc(Br)c([N+](=O)[O-])c1 CCC(CC(=O)NCCC1(CNC(C2CC3C=CC2CC3)=O)CC1)C(C)C c1(C(N(CC(C)(C)CNC(C23CC(F)C2C3)=O)C)=O)cnc2ccc(F)cn12 c1(C(=O)NC2C(NC(C(C)(C)C(N)=O)=O)CCCC2)cnn2c(=O)cc[nH]c12 Cc1cn2nc(N3CC4(CCN(C(c5cc6cccn6cn5)=O)C4)C3)sc2n1 C(C(=O)N1CCCC1(C)NC(=O)CCOc1ccc(OC)cc1)(C(C)C)OC c1(C(N2CC(C)C(NC(c3ccsc3)=O)C2)=O)cnn2c1NCCC2C(C)(C)C C(C)(C(C)(C)C(=O)NCCC(O)CCO)NC(CN(C(=O)OCC)C)=O N1(C(CC2N(C(C(C)OCC=C)=O)CC2)=O)CC(C)(C)C1COC c1(OC)nc(NC(C)(C)CCNC(C2CCCCC2O)=O)nc(C)c1F N=c1nc(CCC(=O)NC2CC(NC(c3ccc(C(F)(F)F)s3)=O)C2)[nH][nH]1 C1(CC)CN(C(c2cncc(OC)c2)=O)CC1CO c1(NC(c2csc(C3CC3)n2)=O)nc(Br)c(Br)cc1Cl c1(C(=O)NCC2(NC(c3cccc(Cl)c3Cl)=O)CCC2)ccc(Cl)c2occc12 c1cc(-c2nscc2CNCCCn2cncn2)ccn1 C(=O)(CCS(=O)(=O)c1ccccc1)NC1CCCC(NC(C(C)(C)C(F)(F)F)=O)C1 C1(NC(C)=O)CCN(c2ccc(C(=O)O)nc2Br)CC12CCC2 c1(C(N2CC(C)C(NC(c3ccc4c(c3)COC4)=O)C2)=O)cccn2nnnc12 c1(OC)ccc(NC(=O)CNS(=O)(=O)c2cccc(Cl)c2)c2ccoc12 CC1ON=C(C(=O)NC2CCCN(C(C3CC(=C4CCC4)C3)=O)CC2)C1C c1(C(=O)NC(C)CN(C)C(c2c[nH]nc2-c2ccco2)=O)cccc2ccnn12 C1(C#N)(CC(N2CC(CCNC(C3(C)CC(C#N)C3)=O)OCC2)=O)CCOCC1 C1(C(=O)NCC2(F)CN(C(Cc3c(C)n[nH]c3)=O)C2)CC(=O)NC1(C)C Cc1cccc(Cl)c1C(=O)NC1CCC(C)N(C(=O)CCc2ccccc2)C1 CCC(C)CC(C(=O)NCCc1ccc(C)cc1)NC(=O)CCc1cnc(C)o1 c1(NCC(C(C)C)C)[nH]c(=NCCNS(C)(=O)=O)nc2c1cnn2C(C)C N1(C(c2cncc(CC)c2)=O)CC2CC(NC(c3cccc(C)c3F)=O)C2C1 n1(CCNC(C(C)OCC=C)=O)c(C(F)(F)F)nc2cccnc12 c1(C(C)C(=O)N(C)CC2(O)CN(C(C3CCCC3)=O)C2)ccccc1Cl C(CC(=O)NNC(=O)c1cccnc1)c1nccc(C)c1 N1(C(C2C3(CCN(C(c4ccc(O)cc4F)=O)C3)C2)=O)C2COCC1CC(F)C2 N1(C(C(F)=CCC)=O)CC2CCCC2(NC(=O)CCCC(N)=O)C1 C(C)(CC(=O)N1CCC(OCCNC(C2SCCCS2)=O)C1)(C(F)F)N(C)C c1(C(N2CCCC(N(C(C(CO)N(C)C)=O)C)CC2)=O)cccc2ncn(C)c12 CC(C)C(C)(CNC(c1cnc(S)nc1)=O)NC(N)=O.C12CC1CNC2=O N1(C(c2ccc(C(C)C)cn2)=O)CC2CC(NC(C3(Cl)CC3)=O)C(C2)C1 C1(N(C(CN(CC)CC)=O)C)CC2CCC(C1)N2C(=O)CN1C(=O)CCC1=O N1(C(CN2CCCC(CC)C2)=O)CCN(C(C2CC3(CSC3)C2)=O)C(CCO)C1 c1(C(N(C2CN(C(=O)C=Cc3cccnc3)C2)C)=O)cccc2cnccc12 N1(C(CNC(C)=O)=O)CCCC2(CCN(C(=O)CC3CCCCCO3)C2)C1 c1(C(=O)NC2CC(CNC(c3cc(Br)cs3)=O)C2)cc2cccc(O)c2[nH]1 C1(N(C)C(c2cc(C(F)(F)F)cs2)=O)CN(C(=O)C2=NOCC2)CC12CC2 c1(C(=O)NCC(C)CNC(=O)C(c2cncc(F)c2)C)ccc(F)c2c1OCC2 N1(CCCc2ccc(C)cc2)CCC(NC(=O)CCn2c(C)csc2=O)C(C)C1 c1(C(=O)NCc2c(C(N(C3CC(CO)C3)C)=O)scc2)ccc2c(c1)CC2 c1(C(=O)NCCN(C(CC(CC)OC)=O)CC(C)O)cc(F)c(Cl)c(N)c1Cl c1(C(=O)NC(C2CCOC2)CNC(C2(C3CC3)CCCC2)=O)cc(=O)cc(Cl)[nH]1 c1(C(=O)NCC(C)N(C(=O)CCOCCOC)CC)cccc2c1CCO2 c1(OC(C)C)cc(N(S(=O)(=O)CC2(C)CCCCC2)C)c(Br)nc1Br C(=O)(CCC(=O)c1ccc(Cl)cn1)NCC1(F)CC(CNC(C(C)CO)=O)C1 C1(C2(O)CCN(C)CC2)(C(=O)NCC2CCCCN(C(C3(C=C)CC3)=O)C2)CC1 S(=O)(=O)(c1cnn(C)c1)NC(C(=O)NCC1(F)CC(NC(CCCC)=O)C1)C C1(C(N(CCOC)CCNC(C2CS(=O)C2)=O)=O)CCCCO1 C1(C(=O)O)CCN(C(N2CCCC(CCN(C)C)C2)=O)C12CC2 N1(CC(=O)NC(CCNC(C(CC#C)(C)C)=O)C)C(=O)Cc2ccccc2C1=O c1(C(N2CCC(NC(C(C)=C3CCC3)=O)C2(C)C)=O)c[nH]c2nccc-2c1C CC(C)CCC(O)C(=O)N1CC2C(C(=O)NCC(O)C3CCC3)C2C1 C1(NC(c2cccc(OC)n2)=O)CCN(C(=O)C(=O)N=S(C)(C)=O)CC(C)(C)C1 N1(C(C(N2CC(C)C2)C)=O)CCC2CCCC12C(=O)NCc1ncco1 N1(C(C(CC(C)C)O)=O)CCC(C2CCCN(C(c3cccn3C)=O)C2)C1 CCCC(CC)C(=O)N1CCN(C(c2cnc(N(C)C)cn2)=O)CC1CC1CC1 N1(C(CCCCSC)=O)CCCN(C(c2cc(C3CC3)ccn2)=O)C(CO)C1 CC1CN2CCN1CC2C(=O)NCC1CC2(CC2)CN1C(c1cnn(C)c1N)=O C(=O)(C(O)(C(C)C)C(F)(F)F)N1CC2CN(C(c3ncc(C)nc3)=O)CC2(C)C1 C1(C(=O)NCCC(CCC)O)CCCCCCN1C(=O)CSC S(=O)(=O)(c1cccnc1NC(C)CN1CCCC(C)C1)N(CCC=C)C CCC(CCC(=O)N1CCCC(O)C1)NC(C1CC=CCC1C)=O c1(C(=O)NC2C(CNC(C=CCCOC)=O)CCCC2)ccc(F)c(CO)c1 c1(C(=O)NCC(C(C)(C)C)NC(CCCCC=C)=O)ccc(N=S(C)(C)=O)cc1 Cc1nc2c(s1)CCCC2C(=O)NC(C1CN(C(c2cc(C#N)cn2C)=O)C1)C CCCCC(O)CC(=O)N1CCCC(O)(CCNC(c2cc(=O)cc[nH]2)=O)C1 C=CCN=C(NCC(C)C(C)O)N1CCN(c2ccc(C#N)cc2Cl)CC1 c1(OC)cc(C)c(C(=O)NCC2CN(C(c3cccc[n+]3[O-])=O)C2)c(C)c1 N1(C(C(COC)N(C)C)=O)CCN(C(=O)C(C)CC#N)CC(C)C1 C(=O)(CC(CN(C)C)C(F)(F)F)NCC1(F)CN(C(C(c2ccccc2O)C)=O)C1 CCCCCC(C)CC(=O)NC(c1cn(-c2ccc(Br)nc2C)nn1)C c1(CC)cc(C(=O)NC2C=CCN(C(c3ccc(C)c(O)c3)=O)C2)ccc1C N1(Cc2cc(OC)cc(Br)c2)CCC2(CCN(C(c3cc(C)oc3C)=O)C2)CC1 c1(OC)c(C(=O)NCC(C(C)C)NC(C2CCCCC2C(N)=O)=O)cnn1C c1(OC)cccc(CC(N2CCCCC2CNC(=O)Cc2cc(C)on2)=O)c1 c1(CC(=O)NC2CCC2CNC(=O)CC2(C3CC3)CC2)ccc2nc[nH]c2c1 N1(C(C2CCC(C(N)=O)CC2)=O)CC2CCC1CN2C(c1cscc1Cl)=O N1(C(CC(C)C(F)(F)F)=O)CCCC2(NC(c3ncc(F)cn3)=O)CCCC12 C(C(=O)NOCC(O)C(C)C)(C1CC=CCC1)NC(c1cc(C(C)=O)oc1)=O N1(C(CC2(C)CCCO2)=O)CC2(NC(c3ccc(O)c(F)c3)=O)CCCC2(F)C1 N1(C(C(C)Oc2ccccn2)=O)CCOCC1CNC(=O)Cc1ccc(O)nc1 c1(SC)cccc(NC(=O)CC2(C)CCN(C(c3nc(Cl)cs3)=O)C2)c1 N1(C(c2cn(C)nc2)=O)CC(NC(c2cccc3c2NCC3)=O)CC2(CCC2)C1 c1(OC)c(F)cc(Cl)cc1S(=O)(=O)Oc1cc(C)cc(Br)c1 S(=O)(=O)(c1ccc(NCC2CC2C2CCC2)cc1Cl)NCCN1CCCC(C)C1 C(C)(N=c1[nH]c(=NC2CCC(C)(C)C2)[nH]c2ccsc12)c1scc(C)n1 N1(CCS(C)(=O)=O)CCOC(c2noc(C3CCCC3)n2)C1.C(=O)(CC1CC1N)N c1(C(N2CC(CC)C(C(=O)NCCC3CCCC3(C)C)C2)=O)cccc(F)c1N C1(C(=O)NCC(CCOC)NC(c2cc(CC)ncn2)=O)CCCC2(CCC2)C1 c1(C(N(CC(CC)NC(C2(C(C)C)CCCO2)=O)C)=O)c(C)cnc(OC)c1Cl CCCC(CCCNC(=O)C=Cc1ccc(CC)o1)NC(C1CCCCCC1)=O C1(N(C(COC)=O)C)CCCC2CN(C(c3cnn(C(F)F)c3)=O)CC12 N1(C(c2cccc(C#C)c2F)=O)CCN(C(C2CC2(C)C)=O)C2CCCC12 C12(C(NOCC(CC)C)=O)COCC1CN(C(=O)C(C)(C)CC(C)C)C2 C1(C)(NC(CNS(CCCC)(=O)=O)=O)CCC(NC(=O)Cc2ccn(C)n2)CC1 c1(C(=O)NC2C(CNC(CCOCC)=O)COC2)cc2cnccc2[nH]1 C1(C(N2CC(OC)(CNC(C3CC4CC3C3CC43)=O)C2)=O)CN(C)CCN(C)C1 n1(CC)cc(Cl)c(C(=O)NC2CC(C)N(C(=O)Cn3cnnc3)C2)n1 C1(C(C)C)(C(=O)NCC(C)(O)C(F)F)CCN(C(=O)Cc2nccn2C)C1 Cc1cc2nc(N3CC4CCC3CN4C(c3cncc(Cl)n3)=O)cc(=O)n2o1 CN1CCC(C(=O)NC(CCC2CC2)C(=O)NC2CC(Cl)(Cl)C2)CC1=O C(=O)(C#CC1CCOC1)Nc1cc(C(NOCC)=O)c(F)cc1 C1(NC(C2CCC(C)(C)OC2)=O)CCC2(CC1)CC2NC(=O)COC1CCC1 CC(C)C(C(c1ccccc1)NC(=O)NCC1CC1)NC(C12CC3CC1C2C3)=O CC1C(C(=O)NC2(c3nc[nH]n3)CCC2)CCN1C.C1C(=O)NCC=CC1 N1(CC(=O)NCC2CCN2C(=O)COCc2cccnc2)CCOCC1=O c1(-c2cn(C3C(OC)CCOC3)nn2)cc(C)c(Br)cc1C c1(OC(C)C)ccc(NC(=O)CSCC2CCCC(C)O2)cc1 N1(C(c2ccc(C(=O)OCC)s2)=O)CCN(C(=O)C(C)C(O)CC)C(CF)C1 C1(CNC(=O)CCC2CC2(Cl)Cl)CC2(CCN(C(=O)C(F)(F)CC3CC3)C2)CO1 Cc1c(Cl)ccnc1C(=O)NCC(C)CNC(=O)CCCc1nncn1C c1(CNCC(C(C)C)(C)O)ccc2cc(C(=O)O)[nH]c2c1 c1(SC)ccc(OCC(=O)NC2CCCC(NC(C3CC(=O)N(O)C3)=O)C2)cc1 c1(C(N2CCC(NC(CCC#CC)=O)C2C)=O)noc2c1CCc1ccccc1-2 C(=O)(C(C(C)C)NC=O)NC(C(=O)N(C(CC)CC)C)c1ccoc1 c1(C(N(CCOCCNC(c2n(CC)ccn2)=O)C)=O)ncccc1CO c1(OC)ccc(C(N2CCCC2CC(N2CCC(O)C(C)C2)=O)=O)c(Br)n1 C1(CNC(C(C)=CC)=O)CCC(NC(=O)CCNC(c2ccco2)=O)C1 c1(NC(Cc2cc(C)on2)=O)c(C)cccc1C.C12CCN(C1)CC(=O)N2C1CC1 C1(C(=O)NCC(=O)NC)COCCN1Cc1ccccc1-c1ccccc1C Cc1snnc1C(=O)NC(C1(NC(=O)CN(C)C(C)C)CC1)C C1(C#N)(CNC(C2C(OC)CN(C(=O)CCC(=O)C3CC3)C2)=O)CCOCC1 c1(C(=O)NCC(CNC(C2C(OC)(OC)CC2)=O)O)cc(=O)c(Br)c[nH]1 N1(C(c2cc(OC)ncn2)=O)CC(O)C(O)C1CNC(=O)C(C)S(N)(=O)=O C(=O)(C(C)C(C)NC(=O)CCCOC(C)C)N(CCCC)CCOC CCCCCC(C)NC(=O)C(CCC1CCC1)NC(=O)CN1CCC(C)CC1 c1(C(N(C)CC2CN(C(CN3CC(C)C3)=O)CC23CC3)=O)cccc(S(C)=O)c1 C1(O)(C(=O)NC2(CNC(c3nn[nH]c3Cl)=O)CCC2)CCCc2ccccc2C1 c1(C(N2CCC(C)(C(=O)Nc3n(C)nc(Br)c3)C2)=O)ccnc2ncccc12 n1(CC)cc(C(=O)N(CCC(C(C)C)NC(C2CCC(=O)O2)=O)C)c(C(C)C)n1 CC1CCCC=C1C(=O)N1CC2CCC2(CNC(=O)C=Cc2ccco2)C1 N(C1CCc2cccc3cccc1c23)C(N(C(c1cccc(F)c1)CO)C)=O N1(C(COCCOC)=O)CCCC(C)(O)C1.C123CCCC1(C2)C(=O)N3 N1(C(Cc2c(C)ccs2)=O)C2CCC1CN(Cc1cccnc1)CC2 c1(CC)ncc(C(=O)NC2CCCC2NC(=O)C(C(C)C)OC)c(O)n1 Cn1nnc2c(C(N3CC(C4CN(C(=O)C5=CCCCCC5)C4)C3)=O)ccnc12 CC1CN(C(=O)Cc2ccn(C(F)F)n2)CC1Nc1cc(C(N)=O)ncn1 N1(C(c2ccc(C#C)cc2C)=O)CCC2CCC(C1)N2C(C1(C(C)C)CC1)=O CC(C)C(C(=O)NC1CCC1NC(c1ccccc1C(C)(C)C)=O)n1cccc1 CC(CC(=O)N(C1(CC(=O)N(C)CC2CCCCC2)CC1)C)CC(C)(C)C C(=O)(C1CCCc2c[nH]nc21)N1CCC(NC(c2ncn(C)c(=O)c2)=O)C1 N1(CC(=O)N(CCCC)C)CC(F)(C(=O)O)C1 c1(CN2CCN(CCCNC(C3CC(=O)C3)=O)CC2)cccc(O)c1Cl c1(C(=O)NCC2(F)CC(CNC(=O)C(O)C3CC3)C2)cnc2n1CCS2 C1(C(=O)NCCNC(C23CC(C)C2C3)=O)CCCN(C(c2ccc(F)o2)=O)C1 CS(=O)C1CN(C(=O)CCN(C(C2CC2F)=O)CC2CC2)C1 Cc1c(C(=O)NC23CCC(CN(C(=O)CCC(C)(C)C)C2)C3)[nH]c2ccccc12 C=C(C)CCCC(=O)N1CCC(N(C(c2[nH]cc(C)c2C)=O)CC2CC2)C1 CC1(NC(c2cnc(Cl)cn2)=O)CCN(C(c2snnc2C2CC2)=O)C1 C1(O)(CNC(Cc2ccc(C(C)C)cc2)=O)CCCN(C(=O)C(C)N2CCC2)C1 Cc1cnn(C)c1C(N1CCC(C(=O)NC23CC(F)(C2)C3)C1C(C)C)=O c1(CCC(=O)NC(CC)CNC(C2CCCCS2)=O)cccc(OC)c1F C(CC(F)F)(C(=O)NCc1oc(C)nc1C)N(C(CCNC(=O)NC)=O)C N1(C(c2c(C)nccn2)=O)CC(NC(=O)CCc2nncs2)CCC1C C(=O)(C(C(C)O)NC(=O)C1CC1)NC(CNC(Cc1ncc(C)s1)=O)C C1(NC(CC(=O)OCC)=O)C2CCC1CN(C(c1scc3c1CCCC3)=O)C2 CC1CNC(C)CN1C(=O)C(C)(F)c1ccon1 c1(C(N2C(CCNC(Cc3c(C)ccs3)=O)CCCC2)=O)ccn2nccc2c1 C(=O)(C#CC1(C)CCCO1)NC1C(C)(CN(C(c2c(CC)nn[nH]2)=O)C)CCC1 N#Cc1cc(CN2CC(CNC(c3c(Cl)cccc3Br)=O)C2)ccc1F C1(NC(c2cc(CC)no2)=O)COC2(CCN(C(c3nc(Br)c[nH]3)=O)C2)C1 c1(CC(C)C)c(NC)noc1C1CC1.C1CCC(=O)N(C)CCCC(=O)N1 c1(CC)cc(Cl)ccc1C(=O)NCC1CCN(C(=O)CCC#N)C12CC2 C1(NC(C(C)=C2CCC2)=O)CN(C(=O)CC23CCC(CC2)CC3)CCC1C c1(SC(=O)NCCNCC(Cc2ccccc2)N(CC#C)CC=C)ccncc1 O=C1NC2CC(NC(=O)CC3CCCN(C(C4(CCF)CC4)=O)CC3)C(C2)O1 C1(NC(C2C(C)CCS2)=O)CCC(NC(C2(n3ccnn3)CC2)=O)CC1 C1(O)(C(=O)NCC(C2CC2)NC(CCCN(C(=O)OCC)C)=O)CCSCC1 N1(C(C2CCCCN2C(C2CCCC(O)C2)=O)=O)CCC(O)C12CCCC2 C1(=CCNC(C=CCN(C)C)=O)CCN(C(=O)C=Cc2ncc[nH]2)CC1 C1(c2ccccc2)(COC(C)=O)CCN(C(=O)NCCc2ccc(C)s2)CC1 c1(C(N(CCCCCCNC(CC(=C)C)=O)C)=O)c(C(F)(F)F)nc(C)n1O C=C(C)C(C)(O)C(=O)N1CCN(C(c2cc(C3CC3)n(C)n2)=O)CC1 CC(C)(CC#N)C(=O)NCC1(O)CCCN(C(=O)C(F)C2CCCC2)C1 Cc1cc(C(=O)NCCC2CN(C(=O)CC3CCSCC3)CC2C)nc(C)n1 c1(OCC)ncccc1C(=O)NC(C1CCN(C(=O)Cc2cccn2C)C1)(C)C C1(CN2C(COC(C)(C)C(=O)Nc3ccc(Cl)cc3)CCC2)CCCS1(=O)=O C1(CNC(C2(COC)C=CCC2)=O)CN(C(=O)CCN2CCC2)CC1C(F)(F)F c1(CC)cn2c(n1)CC(C(=O)NC1CN(C(=O)C#CC(C)(C)C)CC13CC3)CC2 c1(CC(=O)N(CCCNC(c2c[nH]c(=N)s2)=O)C(C)C)ccc(F)cc1[N+](=O)[O-] C(=O)(C(CC(C)C)CC(C)C)N1C(C)CC(CNC(C2(CC#C)CCCO2)=O)C1 CCCC(CCC)CC(=O)NCC1CC2CCC1N2C(=O)CCC(C)(C)[N+](=O)[O-] C1(CC)CC(O)CC2(CCN(C(c3ncccc3N(C)C)=O)CC2)O1 Cc1cccc2cc(C(=O)NC3CC4CCC(C3C)N4c3nccnc3F)oc12 C1(NC(CC2CC(OC)C2(C)C)=O)CCSC12CN(C(=O)C(C#N)=CC1CC1)C2 CC(C)C(O)C(=O)N(CC1CC(C)(CO)C=CC1)Cc1ccc(-c2nn[nH]n2)cc1 c1(C(=O)NCC(CNC(C2(NC(C)C)CC2)=O)F)nc2c(s1)COCC2 n1(CC(=O)NC2CN(C(C(CCOC)(C)C)=O)CC2C)cc(C#N)c(O)nc1=O N1(c2cn(C)nc2)CC(NC2(C(=O)O)CCC(F)CC2)CCC1=O c1(C2CN(C(c3cc(-c4nn[nH]n4)c[nH]3)=O)C2)ccc(S(=O)(=O)F)cc1 c1(OC(C)C)ccc(Cl)nc1C(=O)NC1CCN(C(C2CCOC2)=O)C1 c1(C(N(CCN(C(CNS(CC)(=O)=O)=O)C)C(C)C)=O)cnc(C)s1 c1(CNC(c2c[nH]nc2-c2ccccc2)=O)ccc(Br)c(C(F)(F)F)c1 n1(C(=O)CCSC(F)F)cccnc1=O c1(NC(C2CCOC2)CC)ccc(S(=O)(=O)N(C)CCn2cccn2)c(Br)c1 CN1CCn2ncc(C(=O)N(C3CC3)CC3CCCN3C(C3CCCCS3)=O)c21 N1(C(C=CC(C)C)=O)CCC2CC2(NC(=O)CCNC(c2cccs2)=O)CC1 c1(C(N(CC(CC)NC(C(CC#C)O)=O)C)=O)ccn2nnnc2c1 c1(C(=O)NC2CCN(Cc3cn(C)nc3O)CC2)cccc2c1OC(C)(C)C2 N1(C(c2c(OC)nccc2)=O)CC2(CCN(C(=O)C(C)C(=O)OC(C)(C)C)C2)C1 c1(C(=O)OCC2(C)CC2(F)F)csc2nccn12 CN1CCN(C(C2CC3(CC3)C2)=O)CC1CNC(C1CCCN1C1CCCC1)=O c1(C(c2n(C(CC)C)nnn2)NCc2ccn(C(C)C)c2)nn(C)cc1C c1(CCC)cc(C(N2CCC2CNC(c2cc(Cl)no2)=O)=O)c(C)o1 C(=O)(CCCCCN(C)C(c1cc(C)oc1CC)=O)N1CCCC(=C)C1 c1(C(=O)NC(C)CCN(C)C)ccc(CNC(=O)CSC(F)(F)F)nc1 C(C)(CCCCNC(=O)CCCN1CCCCC1)NC(CCC=C(C)C)=O C1(CCNC(c2ncn(C(C)C)n2)=O)CN(C(=O)CSCc2cccs2)CCO1 C1(NC(=O)C#CC2CCOC2)CC2CC(C1)CN(C(c1ncccc1Cl)=O)C2 c1(OC)cccc(CC(=O)NC2CCC(NC(=O)CCN(S(C)(=O)=O)C)C2)c1 CC1CN(C(c2ccsc2-n2cnnn2)=O)CCC1NC(C1C(C)(C)C1(C)C)=O C1(N(C(=O)CC2C=CCC2)C)CC2CCC(C1)N2C(C1COC(=O)C1)=O C1(C)(C(N2CC(C)(NC(CC3(NC(C)=O)CC3)=O)C2)=O)CC(O)CN1C Cc1cncc(CCC(N2CC(n3cc(-c4cc[nH]n4)nn3)C(O)C2)=O)c1 N1(C(c2c(NC)cnnc2)=O)CC(NC(=O)Cc2cc(C)n(C)n2)CC(F)(F)C1 c1(C(=O)NC2CCN(C(CNS(CC)(=O)=O)=O)C2)c[nH]c2c(Cl)cccc12 C(=O)(C1=COCCC1)N(C(C(=O)NC1CC2CCCCC12)C1CC1)C Cc1cc(=O)n(C)nc1C(N1CCCCC(NC(=O)C(C2CCCCC2)F)C1)=O CC(C)C(O)C(=O)NCC1(CC(=O)N(CCCO)C)CC1 N1(C(C2(CC)CCC2)=O)CCCC(N2CCN(C(=O)C(C#N)=CC3CC3)CC2)C1 c1(C(=O)NC2(C)CCN(C(C(CCC3CC3)OC)=O)C2)cc([N+](=O)[O-])n[nH]1 O=C1CN(CC(C2CCOCC2)C2CCCO2)C(=O)N1CCn1cc(Br)nn1 Cc1cccc2c(C(N3CCCC3C(C)NC(c3ccncc3)=O)=O)cccc12 c1(C(N(C2CCN(C(COCC#C)=O)C2)C)=O)ccc(-c2nnc(O)n2C)cc1 C(=O)(NOCC(F)F)NCC(c1ccsc1)C c1(N(C)CC)cccc(COCC(c2ccc(-c3cccs3)cc2)CC(=O)O)c1 C1(OC)COCCC1CC(=O)N(CCCNC(=O)CCc1ccsc1)C1CC1 c1(OC)cccc(C(=O)NC2CCN(C(c3cc(Cl)c(Cl)n3C)=O)C2C)c1OC C1(NC(c2c(C)c(C3CC3)on2)=O)CC2CCC(C1)N2C(=O)CCC(C)(C)C O(N1C(=O)c2ccccc2C1=O)C(=O)CNC(CCNS(N(C)C)(=O)=O)C(=O)O c1(OC)ccc(-n2cccc2)c(NC(=O)Nc2ccccc2CF)c1 c1(OC)ccc(CN2CCCC(F)(CNC(=O)CC3CCCCC3)C2)c(OC)c1 N1(C(C(COC)NC(=O)OC(C)(C)C)=O)CCCN(C(=O)C(Cl)=CCl)CC1.C(C)(=O)O c1(C(=O)NC)cccc(C(=O)NCCOC2CC(CNC(=O)C(C)(C)OC)C2)n1 CCC(C)C(C)CNC(=O)C(c1cnn(C)c1)NC(=O)CC1CCCNC1=O C1(CC)CN(C(c2cnc(OC)c(Cl)c2)C(=O)NC(C)C(=O)OC(C)C)C(C)CO1 C1(C(=O)NC2CC(CO)C2)CSCCN1C(=O)C1CC1 C1(C(=O)NCCOCC)CC2CN(C(C3(F)CC=CCC3)=O)CC2C1 C(=O)(C(N)C(=O)N1CCN(C(C#N)C#N)CC1)OCC S(=O)(=O)(CCC(=O)NCC1CCCN1C(c1nocc1Cl)=O)NCCNC(C)=O CC1CCC(CCNC(C2(N(C)C(c3cc(C4CC4)on3)=O)CC2)=O)O1 c1(C(=O)NC2(CC=C)CCN(C(=O)CCCCF)C2)cccc2nc(O)ccc12 C1(CNC(c2n(CC)cnn2)=O)CC2CCC1N2C(c1ccc(Cl)nc1N)=O C1(C(=O)NC(CNC(C2C(CC)C2)=O)CO)(SC)CCN(C)C1 CCCCCCC(CC)NC(=O)CC(C)(C)CNC(c1cc(O)ccc1F)=O c1(CC(=O)NCCN(C(c2csc(Cl)n2)=O)CC)ccccc1OC c1(OCC)ccc(C=CC(=O)NC2CC2NC(=O)C(C)=C(C)C)cc1OC C(=O)(C#CC1CCCC1)N1C(C)CC(CNC(CCc2onc(CCC)n2)=O)C1 O=[N+]([O-])c1cc(Br)c(F)cc1CC(=O)Sc1nnnn1-c1ccccc1 N1(C(C2=C(C)C(C)(C)OC2=O)=O)CCCC(C2CCN(C(=O)C(C)(F)F)CC2)C1 C1(n2cccn2)(OCC)CCN(C(=O)CSc2cccc(C(F)(F)F)c2F)CC1 N1(C(C(CC=CCC)C)=O)CCCOC(CNC(c2cnc(N(C)C)s2)=O)C1 C12(C(=O)NCC3CC(NC(CNC(C)=O)=O)C3)CC(C)(C1)C(c1ccccc1)O2 C1(CN2C(C(C3CC=CCC3C(F)(F)F)=O)CCC2)CCCCCC1 c1(C(=O)NC(c2ccccc2F)CNC(C(C)CO)=O)ccccc1N=[N+]=[N-] C(CCC)(C(=O)N1CCCC1C=CC(N1CCC(C(=O)NC)C1)=O)=CCC C(C)(CC(=O)NC1CCN(C(=O)CCc2ccoc2)CC1)(C(F)(F)F)N(C)C N1(C(c2ccc(CSC)o2)=O)CCC(NC(C2CC=CCC2)=O)C(C)C1 c1(C(=O)NC(CN(C(c2ccnc(C)c2)=O)CC)C)ccc(F)c(C)c1N C1(C(=O)NCC2CC2CNC(C2CC=CCO2)=O)(CC)CCOC1 c1(C(=O)NC2C(C=C)CN(C(=O)CSc3cccs3)C2)ccc2c(c1)CCO2 C1(C(N(CCCN(C(CCN(CCOC)C)=O)C)C)=O)CCCC(OC)C1 C(CC(CO)C(C)C)NC(c1c(C)nc(CNC(c2ccc(C#N)[nH]2)=O)o1)=O c1(OC)cc(OC)c(CNCC23CC(C2)C(CC(=O)N)O3)cc1N.C(C)(C)(C)O C1(OCC=C)CCN(C(=NCC(=O)N(C)C)NCC2(C)CCCC2N(C)C)C1 CC1CN(C(c2csc(C3CCCCC3)n2)=O)C(C)CC1C(=O)O N1(C(C2N(C(C(CC3CC3)OC)=O)CCC(C)(C)C2)=O)CCC2(CNC(=O)C2)C1 N1(C(C(c2cccc(F)c2)C)=O)CCC(NC(=O)CC2COC(=O)C2)CC1 c1(NC(CN(C(=O)CCC2CC2)CCOC)=O)cc(C)cc(C#N)c1 C=CC(F)(F)C(=O)NCC1CCN(C(c2cn(Cc3ccccc3Cl)nn2)=O)C1 CN1CCCC1CC(=O)NCC(C)(O)CNC(=O)CCc1cnc(C2CC2)o1 Cc1c(Br)ccc(C(=O)NC(C)C(C)NC(c2ccc([N+](=O)[O-])n2C)=O)c1N C1(CC(N2CC(CNC(C(C)NC(N)=O)=O)C(C)C2)=O)CCCC2(CC2)C1 CC1CN(C(=O)NCCc2cc(O)ncn2)CCN1C N1(C(C(=O)NCC(C)C)c2ccsn2)CCCCC1C1CCC1 C1(C)(C(=O)NCC(C)(C2CC2)NC(=O)C(=O)NCC2CC2)CCCNC1=O N1(C(c2cc(C)cc(O)c2)=O)CCC(C2CC2)C1C(=O)NCCCSC(F)F O=C(C1=COc2ccccc2O1)NCCOC1CCN(C(=O)CCC2CCC2)C1 C(=O)(C1CC(=O)Nc2cc(F)ccc21)OC(C(C)C)C(=O)N1CCN(C)CC1 C1(CC)CN(C(c2cc(C)nc(O)c2)=O)CCC1CNC(C1COC(=O)N1)=O c1(C(=O)OC)cnc(C)c(C(=O)N(C(c2ccc(F)cc2)C(N)=O)C)c1OC c1(C(C(=O)NCC(CNC(=O)C2=CCCC2)OC)O)ccc(Cl)cc1 N1(C(c2nc(NC(C)=O)sc2)=O)CCCC(C)(CNc2nncs2)C1 C(C)(CO)(C(=O)N(CCC(=O)N(C)CC1CCN(C)CC1)C)OC c1(N2CCCC(OCCOC)C2)ncc(C)cc1S(=O)(=O)NC(C1CCCO1)CO Cn1ccnc1S(=O)(=O)N1CCN(C(=O)C(=O)NCC(=O)NC2CC2)CC1 C1(N(C2CCCCC2)C2(c3n(C4C(F)C4)nnn3)COC2)CC2(CCCCC2)C1 C1(NC(=O)C2CC2)CC(NC(C2CC2c2cccnc2)=O)C(O)C1 C1(NC(CCOCCOC)=O)C2CC1CN(C(C1CCC(O)CC1)=O)C2 C1(CCC#C)CCCN(C(=O)CCN(C)C(c2cc(CC)ccn2)=O)C1 C(c1ccc(F)cc1F)=CC(=O)NCC(C)N(C(c1nnc(O)cc1C)=O)CC c1(C(=O)NC(C(CO)NC(C(CC)SC)=O)C)sc(C(C)(C)C)nc1C N1(C(CC2N(C(C(n3ccc(C)n3)C)=O)CC3(CC3)C2)=O)CCn2nncc2C1 C1(CC)CN(C(c2cn(C(F)F)cn2)=O)CC1NC(c1cc(OC)n[nH]1)=O C1(CNC(C2N(C)CCC2)=O)(CNC(c2ccnn2C2CCC2)=O)CC12CCC2 C(=O)(C#CC(C)(C)C)NC(CCOCC)C(=O)N(C)Cc1c[nH]nc1C C1(CNC(C(C=CCCC)O)=O)CC2(CC2)CN1C(=O)C.c1(C)nc[nH]n1 C(=O)(C(CCC1CCC1)NC(c1csc(=N)[nH]1)=O)NC(C)C(=O)NC(C)(C)C C12(NC(C3CC(C(C)C)C3)=O)CCCC1N(C(=O)CC1CCCC1)CC2 c1(OC)cc(C)c(C(N2CCCCC(NC(=O)C3=C(C)OCC3)C2)=O)c(F)c1 C1(C)(Cc2ccc(F)cc2)CCN(C(=O)NC(CC#C)Cc2ccccc2)C1 c1(CNC(CS(CC)=O)=O)cc2n(n1)CCN(C(c1coc(COC)n1)=O)C2 C1(O)(CCNC(C=C2CCN(C)C2)=O)CCN(C(C2(C)CC=CC2)=O)C1 Cc1c(C(N2CCC(C(=O)NCCOCC3CCCC3)(CF)C2)=O)nnn1C c1(C(=O)NC(CC(C)C)CNC(=O)C=Cc2ccncc2)nnc(O)cc1O Cc1c(C(N2CCC(NC(=O)CC3CCC(=O)N3)C2C)=O)cnn1CCO C(=O)(CC(F)(F)C(F)(F)F)NCC1N(C(C2NC(=O)C(F)C2)=O)CCC1 N1(C(C2(C(N)=O)CCC2)=O)CCC2(CC(NC(=O)CC34CC(C3)C4)CO2)C1 c1(C(C)C)n[nH]c(=NCC2CC(NC(c3cnc(Cl)[nH]3)=O)C2)o1 C(N=c1nc(-c2ccccc2)[nH]c(=NC2CC(C)(C)OC(C)(C)C2)[nH]1)C1CC(C)C1 c1(SC)cc(Br)ccc1C(=O)NCCC(C)CCNC(=O)CNC=O C(=O)(C(CO)c1ccccc1)NCC(CNC(C1(C(=O)OC)CC1C)=O)C N1(C(C2=C(C)OCC2)=O)CC(C)CN(C(c2csc(Br)n2)=O)C(C)C1 c1(C(=O)NCC(C(C)C)NC(=O)C2=NOC(C)C2)cc(Br)c(F)cc1Cl c1(CC)cc(F)c(C(=O)NCCCN(C(=O)COC2CCCC2)C2CC2)c(F)c1 c1(CC)cc(C(=O)NC2CN(C(=O)C=C3CCCCC3)C3CC23)ccc1Cl c1(COC)ccccc1NC(=O)C(F)C1CC(NC(c2cc(C3CC3)no2)=O)C1 Cc1ccc(O)cc1C(=O)NC1CN(C(=O)CC(=O)N(C)C)CCC1C(F)(F)F c1(C(N2CC(C(C)NC(C(C)=CC)=O)OCC2)=O)ccc(-n2cccc2)nc1 CCC(C)(C(=O)NCC1CC(NC(=O)C(Cc2ccc(F)cc2)OC)C1)OC C(=O)(CC(C)(O)COC)NCCCN(C(=O)C1=CCN(C)C1)CCC c1(C(=O)NC2C(C)N(C(=O)CN(C)C)CCC2)ccc(P(C)(C)=O)cc1 C12(C(=O)NCC(C)NC(=O)CC3CCC4CC3C4(C)C)CCC(C)(CC1)OC2 C1(NC(CNC(c2c(C)occ2)=O)=O)CCC(NC(=O)CC2NC(=O)NC2=O)CC1 N1(C(c2c(C)nco2)=O)CC(C)(C)OCC1CNC(c1c[nH]c2ccncc12)=O C12(NC(c3cc[nH]c3C3CC3)=O)CCN(C(=O)Cc3cc(F)cc(F)c3)CC1C2 c1(OC)ccnc(CNC(=O)C(C(C)C)NC(c2ccoc2Cl)=O)c1 c1(C(N2CCC(N(C(C3C(C)C3C)=O)CC)C2)=O)ccc2c(c1)N(C)C(=O)C2 C(CC1CC1)(CC(=O)NC(CC1CCC1)CO)NC(c1c(C)n[nH]c1)=O CC1(C)C2CCC1(C)C2C(=O)NC12CC(C1)N(C(c1cc(Br)cnc1O)=O)C2 C1(CC(=O)NC2CCC(N(C(C(C)c3cccs3)=O)C)CC2)CCCS(=O)(=O)C1 N1(C(c2ncn(C(C)C)n2)=O)CCOC(C)(CNC(=O)C(F)(F)C2CCCC2)C1 c1(C(=O)NCC2(CCNC(C3COCCO3)=O)CC2)cc(F)c2[nH]nnc2c1 C1(CNC(Cc2cc(C)nn2C)=O)CC(C)(C)CCC1NC(C1(N(C)C)CC1)=O CCCCC(CNC(c1cncnc1C1CC1)=O)NC(=O)CC(C)N(C)C C(c1ccc(=N)[nH]c1C)=CC(=O)NCCNC(C(C)Nc1scc(C)n1)=O C(=O)(C(C)(C)C(C)(C)O)N1CCN(C(c2ccc(OC)cc2)C)CC1 C(C)(C(C)(C)C(=O)NCCCCCCN(C)C)NC(C(CC=C)C)=O C(=O)(C1=NNC(=O)CC1)NCC(C1CCN(C(C23CCOCC2C3)=O)CC1)(C)C C1(C(=O)NCC2CCCN(C(C3CCN(C(C)=O)CC3)=O)C2)CC(C)CC(C)C1 N1(C(Cc2c(OC)nccc2)=O)CCC(NC(=O)CC(C)C(C)C)C(F)C1 CC1(C(=O)NCC2C=CCCC2)C=CCN1C(c1ccncc1)=O Cn1cnc(C(=O)NCC2(NC(=O)CCOC3CCCCC3)CCOC2)n1 c1(CC(N2CCC(NC(c3c(C)cc(CC)o3)=O)C2)=O)ccc(C(C)=O)c(O)c1 Cc1cc(CN2CCCCC2c2nnc(C3CCCO3)o2)ccc1Br N1(C(Cc2cn(CC)nc2)=O)CCC(CNC(=O)COCCOC)C(C)C1 Cc1cc(C(=O)NCCCCCn2cc(CCN(S(C)(=O)=O)C(C)C)nn2)cs1 c1(C(=O)NC2(CNC(=O)COC3CC3)CCC2)ccc2c(c1)CCCC2 C1(CC#C)(C(=O)NC2CCCCC2CNC(c2snc(C)c2N)=O)CC=CCC1 N1(C(CCC(C)C)=O)CC(C)CN(CC(C(=O)OC(C)(C)C)C(C)(C)C)CC1C c1(C(=O)NC2CC2c2ccsc2)nnc2ccccc2c1C(F)(F)F C1(CC(=O)NC2(COC)CCN(C(=O)Cc3cncn3C)C2)CCCC(C)(C)C1 c1(C(CNC(=O)Cc2cnn(C)n2)NC(COCC)=O)ccc(OC)cc1 c1(C(=O)NC2CN(C(C3CC(SC)C3)=O)CC2(C)C)ccc2sc(O)nc2c1 C1(C(=O)NCC(C)(CC)NC(Cn2c(CCC)ncc2)=O)CC2CCC(C1)O2 N1(C(COc2c(C(C)C)cccc2)=O)CCC(CNC(=O)COC(F)F)C1(C)C C12CC3CCCC3N1C2=O.c1(C(=O)OCC)[nH]cc(C)c1C(=O)OC.N1CCCC1 CCC(O)C(F)(F)C(=O)NCC1(CC(=O)NC2CCN(C)CC2C#N)CC1 CC12CCC(C(=O)NC3CN(C(=O)Cc4ccc(C#N)cc4)CC3O)(C1)OC2 C1(OC)CN(C)C(C)(C(=O)Nc2nc(SC)c(-c3ccccc3)s2)C1 c1(C(=O)NCC(CC)(C)NC(C2CCS(=O)(=O)N2)=O)ccc(-n2cncn2)nc1 N1(C(CC(C=C)CCC)=O)Cc2ccccc2C1CNC(=O)C(C)CO c1(C(=O)NC)nn(C)c(C(=O)NC2C(NC(C(CC)N(CC)CC)=O)C2)c1Br c1(C(=O)OC(C#C)CC)ccnc(Cl)c1O n12cccc(c1=O)NC(=O)C2.C(=O)(C(C)CC(C)C)N1CC(CC#C)(C(N)=O)C1 C123CCC(CC1NC(=O)CSN(CCOC)C(CC)C(=O)N2)C3.CCO.C1CC1 Cc1ncc(NC(N2CC(F)(F)CC2CC2CC2)=O)cc1C(N)=O C1(NC(CSCC#C)=O)CCCN(C(C2CCC(=O)N2)=O)CCC1 c1(C(N2CCC(CN(C(=O)CC3=CCCC3)C)CC2)=O)cncc(C#N)c1 C12(NC(CN(C)S(N)(=O)=O)=O)CCCC1N(C(=O)CCc1nnc(S)n1C)CC2 n1(C(C)(C)C#N)cccc(NCC(N2CC3CC2C3C(=O)O)=O)c1=O N1(C(C2(C)CCC(C)CC2)=O)CC2CCCN(C(c3cc(Br)c[nH]3)=O)C2C1 Cc1cnc(Cl)[nH]c1=NCC(C)N(C)C(C1CCN(C(=O)N(C)C)CC1)=O c1(OC)ncc(-c2cnc(NC(=O)CCc3ccc(F)c(F)c3)s2)c(OC)n1 N1(C(CSc2c(C)noc2C)=O)C2CCC1CC(CNC(=O)CC=C(Cl)Cl)C2 c1(C(=O)NCC(=O)Nc2c(C)csc2C)cccc2ccccc12 C(CCN=c1c(Cl)c[nH]cc1[N+](=O)[O-])N(C(C1=C(C)CCOC1)=O)C C12(NC(CCOc3c(CC)cccc3)=O)CCCC1N(C(=O)C(O)C1CC1)CC2 c1(C(=O)NC(CC)CNC(C2(C)C=CCCC2)=O)cccc2oc(=N)[nH]c12 c1(C(=O)NCC(CNC(c2cnc(S)[nH]2)=O)OC)coc(C(C)(C)C)n1 c1(CC(N2CCC(O)(CNC(CSCC)=O)C2)=O)cc2ccccc2o1 c1(N(C)CC2CCOC2)nc(=NCC23CCCC2C3)[nH]c2cccc(F)c12 N1(C(COCC=C)=O)CCC(F)(CNC(C2CC23CC(OCC)C3)=O)C1 N#CC1CN(Cc2cccnc2)CCN1C(c1ccon1)=O C1(CCNC(C(C)SC)=O)CCCN(C(=O)CCOc2ccc(F)cc2)C1 Cc1cc(Cl)c(C(N2CCCC(C(C)NC(=O)Cc3ccnnc3O)C2)=O)cn1 Cc1csc(C(=O)NC(C2(C(N3CC(C#N)C3)=O)CC2)C)c1C N(C(=NCCC1CCSC1)NCCNS(C)(=O)=O)Cc1cc(C)ncc1 C1(CNC(C(C)=CC2CC2)=O)CN(C(=O)CCCC(C)C)CC(C)(C)C1 N1(C(C(C2CCN(C(=O)CCOC3CC3)C2)C)=O)CCCC12CCC2 CC(C)C(C)C(C)CC(=O)N1CC2CCCC(C1)N2C(C1CCC2CC2CC1)=O CCCC(C)CC(=O)N1CCN(C(=O)CC2CC=CC2)CC1COC c1(C(=O)NCCCNC(C2CCCC(C)C2)=O)nccc(Cl)c1Cl C1(C)(CC)CCCN(C(C2CC(C)CN2C(c2cn(C)c(=O)cn2)=O)=O)C1 c1(C(=O)NC2COCC2NC(C2CC2C2CC2)=O)cccn2c(CO)nnc12 C1(c2n(CCCOC)nnn2)(NC(C2CCOCC2)C)CCSCC1 c1(C(N(CC(C)(C)CNC(=O)C(n2ccc(C)n2)C)CC)=O)snc(C)c1N CCC(CC(=O)N1CC(CN2CCN(C(c3sc(C)nc3C)=O)CC2)C1)C(F)F c1(C(=O)NC2C(NC(C(CCC)C)=O)CCC2)cc2ccccc2o1 C(C(CC(C)C)NC(=O)Cn1ccc(C(F)(F)F)n1)NC(c1[nH]cc(CC)c1)=O C1(CNC(C2(C)CCC2)=O)CCN(C(C2CC2(c2ccccc2)C)=O)CC1 c1(OC)ccccc1C(=O)C(=O)NC1CN(C(C2CCCCO2)=O)C1 C#Cc1ccc(C(=O)NC(C)(CNC(C2CCC(=C)CC2)=O)C(C)C)c(C)c1 Cc1ccc2c(=NCC34CCC(CC3)C4)[nH]c(=NCC=CCl)[nH]c2c1 C1(CNC(C2C(CC)C2)=O)CCC2CN(c3cc(O)nc(=O)n3C)CCC2C1 N1(C(Cc2cc(CC)no2)=O)CCC2CN(C(=O)CN3C(=O)CCC3=O)CC2C1 C(N=c1[nH]c(N2CC3CC2CN3C2CC2)nc(=N)[nH]1)C1(OC)CCC(C)(C)CC1 c1(CC(N2C(COC)(CNC(C3CNC(=O)N3)=O)CCC2)=O)ccc(Cl)c(C)c1 Cc1csc(C(F)(F)C(=O)NCC(C)(C)CC2CN(C(=O)C=Cc3nccs3)C2)n1 c1(CCNC(C2CCCSC2)=O)c[nH]c2cc(O)ccc12 C12(CNC(c3cc(OC)c(O)cc3)=O)CN(C(C3(C(C)C)CC3)=O)CC1CCO2 c1(C(=O)NCC(c2ccccc2)NC(CNC(CC)=O)=O)cncc(C(N)=O)c1 C(=O)(C(C)P(C)(C)=O)NC(c1cn(CC2CCN(C(=O)C(CC)CC)CC2)nn1)C C1(C(=O)NCC(CCNC(=O)CN(C)S(N)(=O)=O)OC)CCCCC(=O)N1 N1(C(c2ccc(=NCC)[nH]c2)=O)CCCC12CCN(C(C1CC1Cl)=O)CC2 C(CC)(C(=O)N1CCC(C2CCCN2C(=O)CC2CCC(=O)N2)C1)OCC Cc1nnc2ccc(C(N3CCC(CNC(C4C(C)C4C)=O)C34CC4)=O)cn12 C1(C(=O)NCCOC2CCN(C(C3CCC(O)CC3)=O)C2)CCn2cncc2C1 c1(OC)cc(OC)c(C(N2CCCN(C(C3CCC3OC)=O)CC2C)=O)cc1N C12CCCC(O1)NC(=O)NCc1nnc2o1.N1(C(C)(C)C)CCC(=C(F)CO)CC1 c1(C(N(C)CC2CCN(C(c3cn(C)cn3)=O)C2)=O)cc(C#N)cs1 C1(CCNC(c2ccc(CC)[nH]2)=O)CN(C(=O)C(C)(C)CSC)CCCO1 N1(C(CC2(NC(C3CCN(CC)CC3)=O)CCC2)=O)CCOC(C)(CC)C1 c1(C(C)NC(c2cc(C(=O)OC)on2)C)ccccc1N(S(C)(=O)=O)C N1(CC)CCC(CNC(c2sccc2NC(=O)COC2(C)CCC2)=O)C1 N1(C(C(C)O)=O)CC(CCNC(c2cnn(Cc3ccccc3)c2Cl)=O)C(C)C1 c1(C(N2CC(O)(CCNC(c3cn(C)c(=O)n3C)=O)C2)=O)nccn2ccnc12 c1(C(N2CC3=C(CN(C(C4ON=C(C)C4)=O)C3)C2)=O)ccnc2c1cnn2C CCC(COC)C(=O)NC1(CF)CN(C(=O)CCN2CCCCC2C)C1 C1(C(=O)NCCN(CC(C)O)C(c2cn(CC)nn2)=O)CCCC1C1CC1 C(=O)(CCCC(CC)CC)N1C(C(N2CC(CCC)OCC2)=O)C=CCC1 c1(C(=O)N(c2ccc3c(c2)OCO3)Cc2ncc(Cl)s2)cc(Br)c2ccccc2c1 N1(C(c2c(CC)c[nH]c2)=O)CC2CCN(C(c3cn(C(C)(C)C)cn3)=O)CC12 N12CC(C(C)(C)C1)NC(=O)C2.C(=O)(C(C)CC(N)=O)NC(=O)NCC(C)C c1(CC(=O)NC2CC(n3cc(-c4nccc(OC)c4)nn3)C2)ccc(Cl)cc1Cl c1(C(=O)NC2C(CNC(C(F)(F)C3(OC)CCC3)=O)CC2)cncc(C)c1 c1(OC)cc(C(N2CC3CC2C3C(=O)NCc2ccccc2O)=O)nn1C CCCC(C)(CC)C(=O)NCC1CN(C(=O)C=Cc2ccco2)CCC1(C)C c1(C(N2CCCN(CCNC(C3C(C)=CCS3)=O)CC2)=O)nccc2cc[nH]c12 N1(C(C(C(C(C)C)OC)O)=O)CC2CCCC(C1)N(C(=O)CN1CCCC1=O)C2 N1(C(C=CS(C)(=O)=O)=O)CC(NC(c2coc(Cl)n2)=O)C2CCCCC12 C1(C2CCC2)(C(=O)NCC2CCN(c3ccc(Cl)cc3)C2)CC1(F)F CC1(C)CN(C(=O)C(=O)NCC2CC2)CC1CNC(c1ccc(CO)c(F)c1)=O C(=O)(C(CCC)CC(C)C)NC(CC=C)CC(=O)NC(CC(=O)OC)C1CC1 c1(C(=O)NCC(CC)NC(C=CCOC)=O)cn(CCCF)nn1 c1(CSCC)ccc(C(=O)NC2(CO)CN(C(c3csnc3C)=O)C2)cc1 N1(C(CC(CCCCC)C)=O)C2CC=C(C(=O)NC3CCN(CC)CC3)C1CC2 N1(C(=O)CCC2CCCO2)CCC2C(CCN2C(=O)CC2CCS(=O)(=O)CC2)C1 C1(OC)CCCC(C(=O)NC2CCC(N(C)C(c3snc(C)c3N)=O)CC2)C1 Cc1nc(C(C)C)nc(N2CCC(O)(C(C)NC(c3cnoc3)=O)C2)c1Br C1(C(N2C(C(=O)NC3CCN(C(=O)OC)C3)CCCC2)=O)CCC=CCCC1 Cc1cc(CCC(=O)NC(C2(C(=O)NCCCC(=O)N(C)C)CC2)C)on1 C(=O)(NNC(=O)COc1cccc(Nc2cccc(C)c2)c1)C1(NC)CC1(C)C C1(CNC(c2ccn(CC(F)(F)F)n2)=O)C(C2CC2)CCN1C(c1ccco1)=O c1(C(=O)NC2C(C)CN(C(CC3CC(SC)C3)=O)C2)nccc(Cl)c1C c1(C(=O)NC(CCOC)CNC(=O)CNC(=O)C2CC2)cccc(C2CCCC2)c1 c1(CN(C)C)ccccc1C(=O)NCC(O)CNC(c1cc(Cl)cn1C)=O CCC(N=c1nc2ncn(CC)c2c(NCCC2CCCN2C)[nH]1)c1cncs1 c1(N(C2CCCCC2)C)ccc(S(=O)(=O)C2CC2c2ccccc2)cc1 C1(C)(C(=O)NC(C2CN(C(c3cccc(C4(F)CC4(F)F)c3)=O)C2)C)CC2(CC2)C1 N1(C(CCC(CC)C)=O)CC(CNC(c2cocc2C(=O)OC)=O)OC(C)(C)C1 Nc1ncc(Br)cc1C(=O)NCC(CC1CC1)CO Cc1cc2occc2c(=NC(CN(C)C)Cc2ccc(Br)cc2)[nH]1 CCCCCCCCC(=O)NCC(C)CNC(=O)C1=CC2CCC(C1)C2 c1(C(=O)NC(C2(O)CCN(C(C3(O)CCSC3)=O)C2)C)ccccc1[N+](=O)[O-] C1(NC(CCSCC)=O)CC2CC1CN(C(=O)CCN1CCCCC1=O)C2 C1(CC(N2CC(OCC(=O)NC3CCCCS3)C2)=O)CC2C=CC1C2 c1(C(=O)NC)sc([N+](=O)[O-])cc1Cl.N12CCCC(C1)C(C)OC(OCC)C2=O N1(C(=O)NC(c2nc3ccccc3[nH]2)C(C)C)CCC(C#N)(C#N)CC1 C1(C)(CC)CC(NC(c2cnc(OC)c(Cl)c2)=O)CN1C(=O)C=CCOC N1(C(c2ccn3ccccc23)=O)CC2CCCC(C1)N2C(C1C=CCC1)=O C1(C)(CNC(c2c(C)nco2)=O)CN(C(C2(C3CCCCO3)CCC2)=O)CCO1 C(=O)(CC(C)CC(=O)NCC1CCCC1NC(c1cnc2scnc2c1)=O)OC c1(CC(=O)NC(C2CCCN2C(C2CC(C)N(C)C2)=O)C)ccc2c(c1)CCC2 c1(COC)nc(CC(=O)NC(c2cc(C)no2)CNC(c2ccccc2)=O)cs1 c1(OC)ncc(CN2CC(NC(=O)CCN3CCCCC3)C(F)C2)cn1 N1(C(CC)=O)CCCCC1CCCNC(C1CC1C(C)O)=O CCC(CC(=O)NCCSCC(=O)NC1(CO)CCC(C)C1)C(C)C N1(C(c2cnn(CCC)c2C)=O)CCN(C(=O)CSC)CCC1C C1(N(C(c2ccc(CC)o2)=O)CCF)CCCN(C(=O)C(F)(F)c2cncs2)C1 CCCC(O)C(=O)NC(CCC1CC1)C(=O)Nc1ccc(OC(C)=O)nc1 C(C)(C)(CCCC(=O)N1CCN(C2CC2)C(C)C1)NC(c1c(CC)c[nH]c1)=O N1(C(c2c(C)n(C3CC3)nc2)=O)CCC2CCC(C1)N2C(C1CC12CC(O)C2)=O C(CC1=CCOCC1)NC(c1n(CC)ncn1)c1nnnn1CCCF C1(C(N2CC(CC)C(NC(=O)CC3CCCC3)C2)=O)CCOCC12CCCC2 C1(C(N2CCC(NC(C(C)(F)F)=O)C2)=O)CS(=O)(=O)CC(=O)N1 N1(C2CN(C(C(C)CO)=O)C2)CCN(C(=O)CC2(O)CCOC2)CC1 Cc1cccc(C(F)(F)C(=O)N2CC(NC(=O)C(C)NC(c3ccoc3)=O)C2)c1 N(C(=NCc1ccco1)N(C)CCOc1ccccc1F)Cc1ccc(C)s1 C1(CNC(CSCC)=O)CCC2(CCN(C(c3cnc4n3CCS4)=O)CC2)O1 N1(C(C)C)CC(C(=O)NC(CN(C(c2cc(=O)cc[nH]2)=O)CC)C(C)(C)C)CC1=O C(CCN(C(=O)C1=CCSC1)C)(C(C)C)NC(Cc1c(C)ocn1)=O c1(C(N2C(CNC(c3nc(C)oc3)=O)C3CCC2C3)=O)ccc(C)c([N+](=O)[O-])c1 c1(CC(=O)N(C2CCCN(C(c3ccoc3)=O)C2)C)c[nH]c2cnccc12 N1(C(C2(CO)CCN(C(c3nn(CC)c(O)c3)=O)C2)=O)CC(=O)NC(=O)C1 C(C(C(=O)NC(C1CC(NC(C2(CO)CC2)=O)C1)C)OCC1CC1)OC C1(CNC(C(CC)(F)F)=O)CCCN(C(=O)C(C)(C)CC2CC2)CC1 N1(C(C(C(=O)OC)OC)=O)CC(C)CN(C(c2ccccc2OC)=O)CC1C CCCCCC(O)C(=O)NCCOCCC(=O)NCC(C)OC N1(CCN(C(C2OCCC(=O)C2)=O)CCO)CCCC2CCCCC12 CC(C)CC(O)C(=O)N(C1CCCCC1N(C(=O)CCC1CCCC1)C)C C1(CNC(CC=CCC)=O)CCC2(CCC2)C1NC(c1cncc(C2CC2)c1)=O C#CCC(C(=O)NCCc1cscn1)NC(C1CC(C)=NO1)=O CN1CCC(C(=O)NCCN(C(=O)COCC2CCCOC2)C2CC2)CC1=O c1(C(N2CC(NC(C(C)OCCC=C)=O)C(OC)C2)=O)cc(C)c(Cl)cc1C C1(C(=O)NCCC(=O)NC(c2cccc(F)c2)C)CCC(C)(C)OC1 N(C(=NCc1ccc(OC)cc1)NCC1COC(=O)O1)CC(C)(CO)OC N1(C(C)CO)CCCN(C(=O)Nc2ccc(CSc3ccc(Cl)cc3)cc2)CC1 C1(NC(c2cc(OC)nc(Cl)c2)=O)CN(C(c2ccc(O)cn2)=O)CC2(CC2)C1 N1(C(c2cc(CC)c(C)cc2)=O)CC2(CCCC2NC(=O)CCCCCOC)C1 C1(CNC(COCC=C)=O)(COC)CN(C(c2coc(Br)c2)=O)C1 c1(C(=O)NCCC2CN(C(C(CC#C)C3CC3)=O)C2)cc(N)cc(O)c1F N1(C(c2ccc(N)cn2)=O)CCC2(CC1)CN(C(=O)CC=C(Cl)Cl)C2 N1(C(C)C)CCCC(N=c2[nH]c(=NCC(C)(C)N(C)C)[nH]c3c2COC3)C1 CCCCS(=O)(=O)NC(C)C(=O)NCCC(C)NC(c1cnc(C(F)(F)F)s1)=O Cc1cnsc1C(=O)NC(C)CC1CN(C(=O)C=CCn2cncn2)C1 N1(C(CCn2ncn(C)c2=O)=O)C2CCC1CN(C(c1ncccc1Br)=O)C2 c1(CN(CC)CC)ccc(-c2ccc(C(=O)NCC3CCC3)nn2)cc1 N1(C(=O)OC(C)(C)C)CCC2CC12C(N1CC(N2CC(F)C2)C1)=O N1(C(c2c(CC(C)C)onc2)=O)CCCCC(CNC(=O)CC=CC(C)(C)C)C1 CC(C)(CC(=O)NC1CCC1NC(=O)CCCOc1ccccc1)c1cccs1 C=CCC(F)(F)C(=O)NC1CCN(C(=O)CCCc2ncc(C)o2)C(C2CC2)C1 CCC(C)(CO)C(=O)N(C)Cc1cn(C2CCN(C(=O)OC(C)(C)C)CC2)nn1 CCCC(C)(CC)C(=O)NC1CCCN(C(=O)COc2cccc(F)c2Cl)C1C c1(C(N(CCC2N(C(CC(C)O)=O)CCCC2)C)=O)ccc2c(c1)NC(=O)C2=O C1(NC(C2C=CC(CC(=O)N(C)Cc3cn(C)nn3)C2)=O)CCCCCCC1 Cc1nc(C#N)cc(=NCCC(C)NC(=O)C(C)CSC(F)(F)F)[nH]1 c1(CC)cncc(C(=O)NCC(C)(O)CNC(c2cc(C3CCC3)no2)=O)c1 N1(C(CC(C)OC)=O)CC2(C1)CN(C(=O)Cc1ncn(C)c1C)CC2CO C1(C(N(CC#C)CC)=O)CC2CC1CN(C(=O)C1=CCC(C)CC1)C2 C(=O)(C(C)(C1CCC1)NC(=O)C(C)OCC)NC(CC#C)C C(C)(C12CC3CC(CC(C3)C1)C2)=CC(=O)NC(CNC(C(CC)F)=O)C C1(C(=O)Nc2cccc(C)c2)CC2CN(C(=O)CCC3CCCOC3)CC2C1 O=C(CC1CCc2cc(Br)ccc21)N1CCCN(C(=O)C(O)C2CC2)CC1 N1(C(C=CCOCCOC)=O)CCCN(C(c2c[nH]c(=N)o2)=O)CC1C C1(CCNC(c2c(OC)nsc2)=O)COCCN1C(=O)CC1CSCCO1 C1(NCc2c(OC)c(Cl)cc(Cl)c2)CC2(CCN(C(=O)OC)C2)CO1 C1(CCC)CN(C(=O)C=CCCC(C)C)CCN1C(=O)C(C)(C)COC Cc1ccc2c(c1)SC(C(N1CCCOC(CNC(=O)CCC3(C)N=N3)C1)=O)C2 N1(C(C(C(CC)O)(C)C)=O)CC2CC(C)N(C(=O)CC3(O)CCCC3)C2C1 C(=O)(C1CCc2cccc(=O)n21)NCC(CNC(c1ccc(OC)nc1C)=O)O C1(OC(C2CCCN(C(c3cccnc3)=O)C2)=O)CC2CCC(C1)C2=O c1(C(N2CCC(C)C(CNC(=O)CCOCC(F)F)C2)=O)cccc2cncn12 C1(S(C)(=O)=O)(C(N2CCC(C(C)NC(=O)CC3CN(C)C3)CC2)=O)CCCCC1 C1(C2CCCN(C(c3ncc[nH]3)=O)C2)(NC(=O)CCc2nc[nH]n2)CC1 C1(C(=O)NCCC)CN(C(=O)C#CC2CCC2)c2ccccc2O1 CC1COc2ccc(C(=O)NC3(C)CCN(C(=O)C(C)CC(F)(F)F)CC3)cc21 c1(C(=O)NCCCN(C)C(C2(N(C)C)CCCC2)=O)cc2n(n1)CCCO2 Cc1cc(=NCCN(C2CCC2)C)[nH]c(NC2CN(C(C)C)C2)n1 c1(C(C(=O)NC(c2ccccc2SC)C(=O)OC)(F)F)cccc(C#N)c1 c1(SCC(=O)OC(C)C(=O)Oc2ccccn2)cc(C#N)ccc1[N+](=O)[O-] Cc1nc(C(C)C)ncc1C(=O)N(C1CC(NC(=O)CCc2ccnn2C)C1)C c1(COC)cc(C(=O)NC2CCC2NC(C2CC(n3ccnn3)C2)=O)n[nH]1 c1(C(=O)NCC(C2CC2)NC(=O)COCCCF)ccc(COC2CCC2)s1 N1(CC(C)NC(COC(C)C)=O)CCN(C(c2cnn(C3CC3(F)F)c2)=O)CC1 N1(C(C(C=C)O)=O)CC(NC(=O)C=C(C)C2CC2)CC1C C1(CNC(c2occ(C)c2)=O)CC2CC(C1)N(C(c1cnn(C)c1C(F)F)=O)C2 N1(CC(=O)NC2CCCC(C(N3CCOC(C(F)(F)F)C3)=O)C2)C(=O)CNC1=O Cc1cc(NC(=O)C(CC(N)=O)NC(c2c[nH]nc2C)=O)cc(CO)c1 c1(C(N(CCCNC(CC2C(OC)CC2)=O)CC2CC2)=O)cc(CO)c[nH]1 C1(CNC(=O)CCOc2cccc(Br)c2)CC2(CC(NC(C3(O)CC3)=O)C2)C1 C1(NC(C=NOC)=O)CCCCCC1C(=O)NC(C)Cc1ccncc1 C=CC(C)(CCOC)C(=O)N1CC(NC(c2nc[nH]n2)=O)C(c2cncn2C)C1 c1(C(=O)NC2CCCN(C(c3[nH]nc(OC)c3Cl)=O)C2)cc2c(cc1N)OCO2 C1(NC(c2cn(CCC)nn2)=O)CC(O)CN(C(C2(CF)CCC2)=O)C1 CCCCCC(=O)NCC(N1CC(CNC(=O)CC#N)C(C(F)(F)F)C1)=O C(CC(=O)N1CCCC1C1CCCC1)(C(F)(F)F)NC(CCCC(OC)OC)=O N1(C(C2(NC(C3CC(F)(CF)C3)=O)C(C)(C)C2)=O)CC2(CCC(=O)N2)C1 c1(C(=O)NC2CCC(CNC(=O)COCC(F)F)C2)cnc2ccc(F)cc2c1 Cn1c(=O)c2cc(C(=O)NS(=O)(=O)CCc3cnoc3)sc2n(C)c1=O c1(C(N2CCC(O)(C(=O)NC3CC(=O)OC3)C2)=O)ccc2ncnn2c1 C(C(=O)NC1CCCC1CF)(C(C)(C)C)NC(c1cn(CC)nc1C)=O C(=O)(C(CC(C)C)c1ccccc1)NC(CN(C(C1(C)CC(=C)C1)=O)C)CC Cc1cccc(-c2cn(CC(C)NC(=O)C(C)C(C)O)nn2)c1 C#Cc1cc(F)cnc1NC(C1CC2CC2N1C(c1cccc(F)c1NC)=O)=O Cc1nn(CC(=O)NCC2CCN(C(C3CCC4(CC4)C3)=O)CC2C)c(C)c1C C12(NC(CCC3(C)CC3)=O)CCCCC1CN(C(=O)CCC(C)(F)F)C2 CC1SCCCC1C(=O)NC(C(=O)NCC1(CO)CCCO1)C1CCC1 c1(C(N2CC(NC(c3ccc(OC)s3)=O)C3(C2)CC3)=O)cc(F)c(C)cc1Cl c1(CCC(=O)NC2C(NC(C(CC(=C)C)C)=O)CC2)ccc2c(c1)CCCO2 c1(OCc2c(OCC)cccc2O)cc(C#N)ccc1C CC1CCCc2nc(C(=O)NCC(CNC(C34CC(F)(C3)C4)=O)C(F)(F)F)cn21 C#Cc1cccc(OCC(=O)NC(CNC(=O)CC2CC3CCC2C3)CC=C)c1 Cc1ccc(Br)c(C(N2CC3(CC3C(=O)Nc3cc(F)ccc3Cl)C2)=O)c1F c1(C(=O)NC2CCC(NC(C(CCC)=CCC)=O)C2)cc(N)cc(OC)c1OC c1(OC)ncc(NC(C2CC23CCN(C(c2ccc(Br)cc2O)=O)C3)=O)cc1F c1(CC)nc(C)c(C(N2CC=CC2CNC(=O)C(C(C)O)N(C)C)=O)o1 c1(C(=O)NC(C)C)ccc(C(=O)NC2CCC(NC(C3(C)CCOC3)=O)C2)cc1 C12C(C1(C)C)C(=O)N2.c1(C(N(C2(CCCCO)CC2)C)=O)coc(C(F)F)c1 C(c1ccc(O)c(O)c1)=CC(N1C(CCCNC(C(COC)OC)=O)CCC1)=O N1(C(c2ccco2)=O)CCC2(CCCCN(C(C3CCC4C(C3)C4(F)F)=O)C2)C1 N1(C(C2(C)CN(C(C3CCN(C)C3)=O)C2)=O)CC2COCC2(C)C1 Cc1sc(O)nc1C(N1CC2C(CC(=O)NCCCN3CCOCC3)C2C1)=O CC(C(=O)NCC1C2CCCC12)C(C)S(C)(=O)=O C=CCN=c1[nH]cc(C(=O)N(C)CC2CCCN2C(=O)C(C)(O)C=C)s1 N1(C(CN)=O)CCn2c(C(=O)Nc3n[nH]c4cccnc34)cnc2C1 c1(OC)cc(F)c(CC(N2CC(CN3CCN(C(=O)C(C)O)CC3)C2)=O)c(Cl)c1 c1(C(=O)NC(C)CNC(c2ccc(C#N)s2)=O)cccc(F)c1Br C1(CNC(CCN(C(Cc2cc(C)on2)=O)C2CC2)=O)CC2C=CC1C2 c1(CC(N2CCCC(c3ncc[nH]3)C2)=O)c[nH]c2cccc(Cl)c12 C=C1CON(C(=O)C2CCCN(C(=O)C(CC)SC)C2C)C1 N1(C(c2cccc(C)c2N)=O)CC(C)(C)CCC1CNC(=O)CCC(C)(F)F c1(C(=O)NC2CCN(CCNC(CC(C=C)C)=O)CC2)nc(OC)ccc1F C1(C(N(C2CCN(C)C2)C)=O)C(C2CC2)CCN1C(c1cc2cccn2cn1)=O CC(C)(C)CCCCC(=O)N1CCC2CCCC12C(=O)NCc1cncc(Cl)c1 N1(C(CCc2c(C)cccc2)=O)CCC(NC(C2C3CCCC23)=O)C2(CCC2)C1 Cc1ncccc1CC(N1CCC2CC12C(=O)NOCCC(C)O)=O c1(-n2cc(CN(C(=O)C(C3CCC3)C3CCC3)C(C)C)nn2)cncc(Cl)c1 C12(C(C)NC(CC3N(C(c4cn(CC)nc4)=O)CC3)=O)CCC(CO1)C2 Cc1c(C(=O)NC(CNC(c2ccc[n+]([O-])c2)=O)CO)nnn1-c1ccccc1 C1(CNC(C2(CCOC)CCCC2)=O)CN(C(=O)Cc2cn[nH]c2)C2CC12 CC(C(=O)NCC1CCN(C(C2CN3CCCC2C3)=O)CC1O)C(F)(F)F N#Cc1ccccc1CNC(=O)COC1CCN(C(C2CCCN2C)=O)C1 C1(C(N2C(C)CC(NC(C3(OC)CCCC3)=O)C2)=O)CN2CCN1C(C)C2 C1(C(N2CC(CN(C)C(C3CCCC3O)=O)C2)=O)Cc2ccccc2N1 c1(C(N2CC(C(C)NC(=O)Cc3cncs3)C2)=O)cc([N+](=O)[O-])n[nH]1 CC1CN(C(C2C3CCC(=O)C23)=O)c2ccccc2N1 C1(CNC(C(=C(C)C2CC2)F)=O)CN(C(=O)Cc2coc(C3CC3)n2)CCN1C C(=O)(C1=CSCCO1)NCC(CCCC)NC(=O)Cc1sc(C(C)OC)nc1C C(=O)(CN=c1[nH]c(C)cs1)NC(CC)CN(C(=O)CCC1CCCCO1)C c1(OC)cc(C(N2CC(C(F)Cn3cc(CSC)nn3)C2)=O)cnc1OC CCC(C)(C)CC(=O)NC1CCN(C(c2cc(C)n(C(C)(C)C)n2)=O)CC1CO Cc1cc(NC(C2(F)CCN(C(c3n[nH]cc3[N+](=O)[O-])=O)C2)=O)c(C)cc1O C1(NC(CN(C2CCSC2)C)=O)(CNC(c2ncc(C(F)F)s2)=O)CCOC1 C(=O)(C(CO)C(C)(C)C)NCC(CNC(CC(C)F)=O)C(F)(F)F N1(C(C(CCC)CC)=O)CC2CCN(C(c3cc(C(C)(C)C)c[nH]3)=O)C2C1 N1(C(=O)CSC(F)F)CCCCC1c1cn(CC2CC3CC3C2)nn1 C1(CNC(CC(C)(C)OC)=O)C2CCCC1N(c1cnc3ccccc3n1)C2 C(CO)(CCCCNC(=O)C1=CCCC1)NC(C(n1ncc(C)c1)C)=O N1(C(C23C(CN(C(C4=CCC(C)CC4)=O)C2)COC3)=O)CCC(C)C(F)(F)CC1 C12(C(=O)NC(c3nn[nH]n3)CC)CCC(NC(c3cnc(C)cc3C)=O)(CC1)C2 N1(C(=O)C=CC2CCOC2)CC2CC(NC(C3(F)CCCC3)=O)C2C1 CCCCC(CNC(=O)C(C)OCOC)NC(=O)CCCNC(C1CCC1)=O c1(C(=O)NC2CCCN(C(C(C=C)O)=O)C2)ccn(CCO)c(=O)c1 S(=O)(=O)(c1ccc(C(=O)NCc2c[nH]nc2C2CCOC2)cc1)NC(CC)C c1(NC(C(=O)NCC(C2CCC(F)(F)CC2)OC)=O)ccc(I)c(Cl)c1 c1(C(=O)OC)nnc(N2CC(O)(C(C)NC(C3CC3C(C)O)=O)C2)s1 C1(C(=O)NC2(C)CCN(C(c3cccc4ncsc34)=O)C2)Cc2ccccc2S1 CCCCC(CC)CC(=O)NC1CCCC1NC(=O)Cc1cccc(OC)n1 C1(CC(=O)NC(C(=O)OCC)C)CCCCC1NC(=O)CCCCSC C1(NC(C2(CCC=C)CN(C(c3cnns3)=O)C2)=O)CCC(C#N)CC1 C=Cc1cncc(C(=O)NCCC(CNC(C2CCSC2)=O)OC)c1 C1(C(=O)NCC(=C)CCNC(=O)CCCNC(=O)NC)CC2CCC(C1)S2(=O)=O c1(C(=O)NCC(C)(CO)NC(CC(C)O)=O)cccc(N2CCCC2)n1 C(=O)(C(F)(F)C(F)F)NCC1(C)CC(NC(C2C(C(C)C)CCO2)=O)C1 C(=O)(CCP(C)(C)=O)NCc1c(C(N2CCCC(C)C2)=O)[nH]cc1 N1(C(C(C)C(C)(C)C)=O)CCCC2(C1)CN(C(c1cc3n(n1)CCO3)=O)CCO2 C=CCC(CNC(c1cn2c(n1)CCC2)=O)C(=O)NC1CCCC2(C1)N=N2 N1(C(c2c(CC)c[nH]c2)=O)CCC(C)(CNC(=O)CC2CC2C2CC2)CC1 c1(SC)cc(C(=O)NC2CC(N(C(=O)COCc3ccnn3C)C)C2)ccc1F n12cc(cn1)C(=O)NCC2.C(C)(CCN(C(=O)CSCCC#N)C)OC CCCC(CCC)C(=O)N1CCC(C)(C)CC1C(=O)NOCCc1ccccc1 C(C(=O)NN1CCCC1C(=O)N(C)CC12CCC(CC1)C2)c1cc(C)sc1 c1(C(=O)NCC(O)CNC(C2CC2Cc2ccccc2)=O)ccc(Cl)cc1O C1(NC(c2cc(C)c(C)o2)=O)CN(C(c2ccc(CS(C)(=O)=O)o2)=O)CCC1C C1(CNC(c2cccc(C)c2)=O)CCCCC1N=c1cc(C)[nH]c(C)c1[N+](=O)[O-] CC1CC(C(=O)NCC2CC(F)(CNC(c3cn4ccnc4s3)=O)C2)=NO1 C1(NC(C(n2ccc(C)n2)C)=O)CCN(C(=O)C=Cc2cn(C)cn2)CC(O)C1 Cc1cc(F)c(C(=O)NCC(C)NC(C2(C)CC(C(F)(F)F)C2)=O)c(F)c1 c1(C(=O)NCCC2OCCN(C(C(C(C)C)N(C)C)=O)C2)cnc2[nH]nnc2c1 N1(C(=O)C(O)(C2CC2)C2CC2)CCOC(c2ncc[nH]2)C1 N1(C(c2cccc(OCC(C)C)c2)=O)CCC(C)C(NC(c2cnc(O)s2)=O)C1 c1(NCC2(O)CN(C(c3c(O)ccc(OC)c3)=O)C2)nc(C)cc(C#N)n1 C1(NC(c2c(C)n(C3CC3)cc2)=O)CCN(C(c2cnc(=N)[nH]c2)=O)C12CC2 C(C(O)(CO)CO)NC(c1nc(CNC(C(C)NC(=O)OC)=O)oc1)=O C1(NC(c2cnccn2)=O)CN(C(=O)CCc2ccc(F)cc2)C2CC12 CC(C)CC(O)C(=O)NCC1CCN(C(=O)CNC(=O)CCc2ccccn2)C1 C12(C)COCCN1C(=O)Cn1cc2nn1.Cc1cc(C(=O)OC(C)(C)C)c(C)s1 N1(C(CN(C(C(=O)NCC(C)NC(=O)OC(C)(C)C)=O)C)C)CCCCC1 C(CN=c1ncc(Cl)c[nH]1)(C1CCCCC1)NC(=O)CCC=CBr N1(C(c2n(C)ncc2CNC(=O)C2=CCCC2)=O)CCC(C)(CO)CC1 C=CC(F)(F)C(=O)NCCN(CC(C)O)C(=O)Cc1ccc(OCC)cn1 C(=O)(CCCCC(N)=O)NCC(C)(C)OCC(=O)NC1C(C)CCCC1 c1(C(N(C(c2cccs2)C)C)=O)coc(CNC(=O)C(N2CCOCC2)C)n1 CC(CN(C)C)CC(=O)NCc1cncn1C.c12ccc-1nc2 CCC(C(=O)OC)C(=O)NCC1C(CNC(=O)Cn2cccnc2=O)C1(F)F c1(C(=O)NCC(CN(C(Cc2c(C)noc2)=O)C)O)csc2ccccc12 CC1=NOC2(C1)CC(C(=O)NCC1CC3(CCC3)CN1C(C1CC(C)(O)C1)=O)C2 C1(CNC(C2(CC(C)C)CC2)=O)CC(C)CN(C(=O)C(C)(C)n2cnnn2)C1 c1(CC(=O)NC2C(NC(C3C(=C)C3C(=O)OC)=O)C2)ccccc1Cl N1(C(C2ON=C(C)C2)=O)CCCC(CO)(NC(=O)C=Cc2ccc(C)cc2)C1 c1(NC(=O)NCCCc2cnn[nH]2)ccc2c(Cl)ccnc2n1 c1(C(=O)NC2C(NC(C(CCOC)OC)=O)CCC2)ccc(F)c2cnccc12 c1(CC)ncsc1C(=O)NC1(CC(=O)NCC2CC2)CC1 c1(CNC(N)=O)ccccc1C1(C(=O)NCC(C)O)CC1.C12(CC1)C(=O)N2 N1(C(c2cc(C)ncn2)=O)CCCCCC(NC(=O)CC2CCCC(C)(C)C2)C1 C1(C(N2CCC(NC(C3(C4CCC4)CC3)=O)C(O)C2)=O)CC2C=CC1CC2 N(C1CC(C)(C)Oc2cc(C)ccc21)CC(=O)NC(CC)(C)C c1(C(N2CCC(O)(CC(C)C)C2)C(=O)NCC(=C)C)nccc2ccccc12 C(=O)(C(C(C)C)SC)NC1CC(CNC(C(C2CCOC2)OC)=O)C1 C1(C(=O)NCCCC(C(=O)OC)O)CC2COCC(C1)C2=O Cc1cccc(C)c1OCC(=O)NC(C)CC(C)NC(C1CC1C#N)=O C1(CNC(C2CC2C(F)F)=O)COCCN1C(=O)Cc1cnccn1 N1(CC(=O)NC(Cn2cc(C3(CC)CCCO3)nn2)C)CCSC(C)(C)C1 C(=O)(CCN(OC)C(=O)CC1(C)CCN(C(=O)CN2CCN(C)CC2)C1)OC c1(NCC2(CCNC(C(C(CC)O)(F)F)=O)CC2)c(C#N)c(=O)n(C)c(=O)n1C C1(C)(CNC(CN(S(CC)(=O)=O)C)=O)CCCC1NC(=O)CC1CCCO1 C1(CC(=O)NC(C(C)NC(c2cnc(-c3ccoc3)s2)=O)C)CCCCCC1 C1(OC)(CNC(C2CCCCC2CNC(c2c[nH]cc2C)=O)=O)CCCCC1 Cc1sccc1CC(N1CC(CNC(=O)CCc2cnoc2)C1)=O Cn1ncnc1C(=O)NCCNC(C1CC1C1CC1)=O c1(CC(C)C)ccccc1-c1c[nH]c(=NCC2CCC(=O)N2)s1 C1(C(N2CC(CCC)C2)=O)(NC(=O)C=CC(F)(F)F)CCCC1C C1(C(=O)NCC2(NC(c3cn(CCCF)nn3)=O)CCC2)(OC)CCOCC1 Cc1c(C(=O)NCC2CCCC2NC(=O)CN2CC(C)C2)ccn1CCO C(=O)(CC(C(F)(F)F)NC(=O)CC=C(Cl)Cl)NCP(OCC)(C)=O N1(C(CCCc2ccc(C)s2)=O)CCN(C(=O)CC2(C)CC2(F)F)C(C2CC2)C1 CC1(C)C(CC(N2CCCCC2CCNC(C2CC3CCC2O3)=O)=O)CC1O C1(F)(CNC(C=C(CC)CC)=O)CCN(C(=O)C(C2CC(F)(F)C2)O)C1 c1(OC)nc(C)ccc1NC(C1CCCCN1C(=O)C(c1ccc(Cl)cc1)C)=O CC(C)(C)CC(=O)N1CC(NC(=O)CCn2cc(Cl)cn2)C(n2cccn2)C1 c1(C(N2CCCC(C)(NC(=O)CC(O)C3CC3)C2)=O)cccc2nsnc12 n1(CC)nnc2c1CCC(C(N1CC(OC)C(NC(=O)CCCC(C)C)C1)=O)C2 C1(C2CCCO2)(C(=O)NCC2(O)CN(C(c3cc(Cl)cnn3)=O)C2)CCCO1 C1(CCNC(c2cc(Br)co2)=O)COCCN1C(C1C2CCCC12)=O c1(NC(N(c2ccc(C3CCCCC3)cc2)C)=O)ccc(F)nc1 n1(CC(=O)N(CCC(C)NC(c2nccc(CC)c2)=O)C)ccc(=O)cc1C c1(CCCC)cc(C(N2CC(CCNC(=O)COCCOC)(OC)C2)=O)n(C)n1 C1(CN(C)C)CC(O)CN1C(c1coc(CNC(=O)C(O)C2CC2)c1)=O c1(OC)cc(C(=O)NCCCN(C)C(c2ccc(C)c(O)c2)=O)c2occc2c1 C1(NC(C2CC(=O)NC2)=O)CCCC12CCN(C(=O)Cn1cc([N+](=O)[O-])cn1)C2 c1(C(=O)NC2C(NC(Cn3ccc(C)n3)=O)CC2)noc2c(F)cccc12 Cc1cc(C)c(NC(=O)CSc2cc3ccccc3s2)c(Cl)c1 n1(CC#C)c(C(N2CC(CNC(c3ccns3)=O)C(C)C2)=O)cc2ccccc12 Cc1ccnc(O)c1C(=O)NCC(C(=O)NC(c1cc[nH]n1)C)C(C)C N1(C(CSCC(C)C)=O)CCC(O)C(NC(C2CC23CCCCC3)=O)C1 C1(C(=O)NC2CC(CNC(c3ccc(C(N)=O)s3)=O)C2)CCCC2(CCC2)O1 CCC(CCCC(=O)N1Cc2c[nH]nc2C1)NC(c1ccccc1OC)=O c1(C(=O)NC(CNC(c2c(CC)c[nH]c2)=O)C(C)C(C)C)nc2c(s1)COCC2 Cc1sc(Br)cc1C(=O)NC(C)CN(C(=O)C(c1ccc(O)cc1)=O)C Cc1cc(C(N2CC(N(C(=O)CCN3CCOCC3)C)C(F)C2)=O)[nH]c1C C12(CNC(N3CCCC3)=O)CC1CN(C(c1ncc(C(=O)C3CC3)s1)=O)C2.C1(N)CC1 C#CC1(C(=O)NCC(C)(COC)CC)CCN(C(=O)C(C)CC2CCC2)C1 N(C1COc2cccc(Cl)c21)C(N1CCCC(CN(C)C)C1)=O N1(CCCNC(CN(CC#C)C(C2CCC2C(C)(C)C)=O)=O)CCCC1C Cc1nc(-c2ccco2)cc(=NCC2CN(C(c3nc(Cl)c(Cl)s3)=O)CCO2)[nH]1 C1(C(=O)NCC2CCCN(C(c3c(CC)sc(=N)[nH]3)=O)C2)CC2(CC(C)=NO2)C1 C(=O)(CC1COCc2ccccc21)N1CCCC(NC(C(C)CO)=O)(CO)C1 c1(CN(C(c2c(C)nc(C(C)C)s2)=O)C)cccc(Cl)c1F.C12CCCN1C2=O c1(C(N(CC(C)C(=O)NCc2nccc(O)n2)C)=O)c[nH]c2nccc-2c1 N1(CCC)CCN(C(C2CCCN(C(=O)COc3cc(C)ccc3)C2)=O)CC1 N1(C(=O)NC(C)(C)C)CC(C(N)=O)CC(C)C1.c12cscc1N(C)C2C(=O)NC c1(OC)c(C(=O)NCCCCC2CN(C(c3cc(C)oc3C)=O)C2)sc(Cl)c1Cl C1(C(N2CCC(F)C(F)C2)=O)N(C(=O)C2=C(Cl)CC2)CC12CCCC2 C(CN=c1[nH]c(N2CCc3nncn3CC2)nc2c1SCC2)C1CNC(=O)O1 Cc1c(C(=O)NCC2CCC2NC(c2cccnc2C(F)F)=O)cncc1Cl C1(C)(C(=O)NCC(C)(C)NC(c2c(COC)cc[nH]2)=O)CCCOC1 C(C(CCO)N=c1nc2scnc2c(NCc2ccc(Br)cn2)[nH]1)OC O=C(C(O)CC(F)(F)F)NCCCNC(C1CC1C(F)(F)F)=O c1(C(N2CC(OC)C(NC(=O)CCNC(=O)CC(C)C)C2)=O)ccc(F)cc1N c1(C(=O)NC2CCCN(C(C(C)=C3CC3)=O)CC2F)ccc(S(N)(=O)=O)c(C)c1 CC(C)P(=O)(CC(=O)NCC1CC1NC(c1cn(C)cn1)=O)C(C)C c1(C(=O)NCC(CNC(C2CC(OCC)C2)=O)O)cnn(-c2ccccc2)c1F N1(C(CCN(C(CC)CC)C)=O)CCC(NC(=O)Cc2[nH]cnc2C)C1 c1(C(N2CCC23CCCC3)C(=O)NC2CCCCC2)cc2ccccc2cn1 C(=O)(C1=C(C)OCC1)N(C1CCC(NC(C=CCC)=O)CC1)C c1(CC(=O)NC2(CCO)CN(C(CCC=C(C)C)=O)C2)cccc2ncccc12 c1(C(=O)NCC(C)(C2CC2)NC(CCOCCOC)=O)cc(C)c(F)cc1N CCCCCCCCCC=CC(=O)NC(CNC(c1cc(C)nc(O)n1)=O)CO C1(NC(CN(C(=O)Cn2cc(C#N)cn2)C)=O)CC2C(NC(=O)C3CC3)C2C1 C1(CNC(C(C)OC)=O)(NC(C2CCCC(C)C2)=O)CCC(C)(C)CC1 C1(NC(Cc2cc(C)on2)=O)CN(C(=O)CCC2CCCCN2C)CC1CO C1(NC(c2cc(OC)n(C)n2)=O)CC2CCC(C1C)N2C(C1(C)C=CCCC1)=O C(=O)(C1=CCCC1C)N1C2C(C(=O)NCC(C)SC)C(C2)C1 C1(CNC(c2cscc2F)=O)CCC2(CN(C(=O)Cc3csc(S)n3)C2)O1 N1(CC(=O)NC2CC(CC(=O)N(C(C=C)C3CCC3)CC)C2)CCOC1=O N1(C(COCC(=O)NC)=O)CC(CNC(=O)Cc2cccn2C)C2CC12 C1(CC(=O)NC2C(CC)N(C(=O)CCC3CCCC3)CC2)CCCC(C)(C)C1 C(=O)(CCS(=O)(=O)C(F)(F)F)NC(C)CCNC(C1CC2CSCC(C1)C2)=O c1(C(N2C(C(=O)NCC(CC)CCO)CC2)=O)ccc(C)nc1C c1(CC)cc(CCCNC(Cc2csc(Cl)n2)C(=O)OC)on1 c1(-c2nc(-c3cccc(C)c3)nn2C2CCCSC2)ccc(Cl)c2cccnc12 N1(C(C2CC(OC(C)C)C2)=O)CCC(C)C(NC(=O)C(F)(F)C2(O)CCC2)C1 N1(C(c2cc(CC)[nH]n2)=O)CCC2C(NC(=O)CC(CC)C3CC3)CC12 N1(C(COCCCOC)=O)CCCC(C)(CNC(C2(C)CC2(F)F)=O)C1 Cc1ccc(F)c(CNC(=O)CC23CCC2CN(C(C2CCCOCC2)=O)C3)c1 C1(CCC)CCN(C(C2(COC)CN(C(=O)C(C)n3ccnc3)C2)=O)C1 C(=O)(CCC(=O)NC(C1CCN(C(=O)C(C)(C)CN(C)C)C1)(C)C)N(CC)CC N1(CC(C)NC(C2(C(F)F)CCC2)=O)CCN(C(c2ccn(C3CC3)n2)=O)CC1 C#CCCCC(C)C(=O)NC(C)(C)C(=O)NC1CC(O)C(O)C1 C12(CNCc3c(SC)cccc3)CCC(C(F)(F)F)(CC1)C2 N1(C(C(CC)F)=O)CCOC2(CCC(NC(c3cc(Cl)sc3Cl)=O)CC2)C1 C=C(Cl)CCC(=O)NCC1C(CC)CCN1C(c1ccnc(S)c1)=O C1(NC(CCNC(=O)C=CCl)=O)CCN(C(C2(CO)CCC2)=O)CC1F c1(CNc2cc(NCC3CC(F)C3)ncn2)ccnc2ccccc12 Cc1nc(S)sc1CC(=O)NCC(C)CNC(c1coc(C#N)c1)=O c1(CN(C)CCN(C(c2cn(CC3CC3)nn2)=O)C2CC2)ccc(=N)[nH]c1 c1(C(=O)NC(CNC(C=CCOC)=O)C(C)C)cncc(-n2cnnn2)c1 c1(CN2CC(C)(N(C)C)C2)cccc2ncccc12 N1(C(COCCC)=O)CCC2(CC1)CCN(C(c1c(C)oc(C)c1C)=O)C2 Cc1ccc(C(=O)NCc2cccnc2CNC(=O)C(C)(C)F)c(Br)c1 C(=O)(C(C)(C)C1=CCN(C(=O)C(C)OC2CCOC2)C1)N1CCCC(=C)C1 CC(C)C(C)C(CNC(c1cc(Cl)cnn1)=O)NC(=O)C#CC(=O)N(C)C C#Cc1ccc(C(=O)NC2CCC2CNC(C2(C(=O)C3CC3)CC2)=O)nc1 Cc1c(Cl)ccnc1C(=O)NC1CN(C(=O)CC(=O)N(C)C)CC1O S(=O)(=O)(CCCCCl)NC(C12CC(NCc3ccn(C)n3)(C1)C2)=O C1(C2CN(C(c3ccc(CS(C)(=O)=O)cc3)=O)C2)(NC(CN2C(C)CC2)=O)CC1 N1(C(C(Cc2ccoc2)NC(c2n(CC)ncc2)=O)=O)CC2CCCC(O)C2C1 Cc1ccnc(O)c1CNC(=O)NC1CCCCCC1F c1(C(=O)NCCN(C(C2C(CC)OCC2)=O)C2CC2)ccccc1-c1cn[nH]c1 C(C1CCc2ccccc21)N(CC(=O)NC)CC1CCC(=O)NC1 CCCCCC(O)C(=O)N1CC(C2CC2)(C(=O)NC(C)CN2CCCC2=O)C1 C(=O)(C(C)OC(=O)CCNC(=O)OC(C)(C)C)OCC=C c1(CC(N2C(C)C(NC(=O)CC3(CO)CC3)CCC2)=O)ccc2c(c1)OCCCO2 C1(NC(CCc2nc(C)c(C)[nH]2)=O)CN(C(c2nonc2N)=O)CCC1F C=CCCC(C(=O)N(CCC(C(C)C)NC(=O)CCCC)C)c1ccccc1 N1(C(C)=O)CCC2CCC(C1)N2C(C1CN(C(C)=O)CCS1(=O)=O)=O.C(C)(C)C C=C(C)CC(C(=O)N1CCC(CN(C)C(C2CC(C)(C)C2)=O)CC1)OC Cc1nc2nccc(N3CC4(CN(C(=O)NC5CCc6ccnn6C5)C4)C3)n2n1 n1(CCCC#N)cc(C(=O)NC2CCCC2CNC(=O)CCn2cncn2)nn1 N1(C(=O)CC2(c3ccccc3)CCC2)CC(NC(C2(F)CCC2)=O)CC1CO N1(C(CC2ON=C(CC)C2)=O)CCN(C(=O)CN(C)S(N)(=O)=O)C2COCC12 c1(-c2nccc(-c3n(CC(C)(C)OC)ccn3)c2)c(C)nn(C2CCOC2)c1C c1(C(=O)NCC(CC=C)NC(c2c(C)ncn2C)=O)cccc(Br)c1N C1(C(=O)NCC2N(C(C3CCC(C)CC3)=O)CCC2C)CC2(CCOC2)C1 C(C(C)(C)C(=O)N(CCC(C)NC(C1CCC(=O)N1)=O)C)OC(C)C C1(C2CCOCC2)(NC(=O)NC2CCN(C(=O)C3CC3)CC2)CC1 c1(OC)ccc(F)c(C(=O)N(C)CCN2CCN(C(=O)C(CO)N(C)C)CC2)c1 C(=O)(C1=CC(C)(C)C1)NCC(C1N(C(=O)CCC=O)CCC1)(C)C.CCN Cc1ncc(CNC(C2CCC(CNC(c3ccccc3)=O)C2)=O)s1 c1(C(N2CCN(c3ncc(F)cn3)CC2)C(=O)NCCC)c(Cl)nc(Cl)n1C C1(CNC(=O)C#CC2CC2)CC2(CO1)CN(C(=O)Cn1cnc(Br)n1)C2 c1(C(C(=O)NC(C)CNC(=O)CSCc2ccccn2)(F)F)cccc(Cl)c1F C1(CNC(c2cncc(NC)c2)=O)CCN(C(c2cc(C)cc(F)c2)=O)C(C)C1 c1(C(N)=O)cc(C(N2CCC(CNC(=O)CCN3CCOC3=O)CC2)=O)ccn1 C1(NC(c2cccnc2O)=O)CN(C(C2CCS2(=O)=O)=O)CC1O c1(NC(=O)CC2CN(Cc3cc(Br)ccc3Cl)CCO2)cccc2[nH]ncc12 N1(C(CCc2cnc(C)s2)=O)CC(NC(=O)C(F)(F)c2cnccn2)C(O)C1 Cn1ccc(=O)c(C(=O)NCC2CC(F)(CNC(C3CCCOCC3)=O)C2)c1 N1(C(C2C(OCC)C2)=O)CCN(C(c2c(Cl)n[nH]c2CC)=O)CC(C)(C)C1 C1(CCC(=O)OCC)CCCN(C(C2(C3CNC(=O)O3)CC2)=O)C1 CCCC(C(=O)NC(C(=O)NC1C2COCC12)C1CCC1)N(C)C C1(CNC(C2(NC(C=CC=CC)=O)CC(F)C2)=O)C2CCCOC12 c1(C(N(C2CCN(C(c3cccc(Br)n3)=O)C2)C)=O)cc2cccc(Cl)c2[nH]1 N1(c2n(CCCOC)c(-c3cc(C)nc(C)c3F)nn2)CCC2(CCC(O)C2)C1 C#CC(CNC(=O)CC1(OC)CN(C(c2cnc(Cl)s2)=O)C1)CC C(C(F)C(=O)Nc1cn(Cc2nccs2)nn1)C1CN(C(CC)=O)C1 c1(C(N(C)CC2(NC(c3cscn3)=O)CC2)=O)cncc(OCC(F)(F)F)c1 C1(c2n(CCC3C(C)C3)nnn2)(NC2COC3(CCC3)C2)CCCSCC1 C1(C(N(C)Cc2ncc(C)o2)=O)CCN(C(C2CC3C=CC2CC3)=O)C12CCC2 C(C(O)(CO)CO)NC(Cn1cc(NC(=O)CC2CCC2(F)F)nn1)=O c1(C2C(C(=O)NC(c3ccc(C)o3)CCOC)C2)nnc(C)o1 CC#CC1CN(C(C2CCCCC2CNC(c2occc2C2CC2)=O)=O)C1 C(=O)(CC1NC(=O)c2ccccc21)NC(C1CC(NC(c2ccnn2C)=O)C1)C c1(C(N(C2CC(NC(C34CC(OC)C3C4)=O)C2)C)=O)ccc2cc(C)oc2c1 Cc1ccccc1OCC(N1CCCC1CCNC(=O)CCc1nccn1C)=O CC(CC(=O)N1CCC1(C)CC(=O)NC1COC(=O)C1)N(C)C c1(C(N(CC(N2CCN(C(=O)CC3(CO)CC3)CC2)=O)C)=O)cc2ccccc2[nH]1 C(=O)(C1=CCC2(COC2)OC1)N1CCN(C(c2c(C)n3c(s2)ncc3)=O)CC1C C1(NC(C(C2CCC2)OC)=O)CN(C(=O)CSCC(F)(F)F)CC1C c1(C(N2CCC(CNC(CC(C)O)=O)C2)=O)cnc2ccccn12 c1(NCC2(F)CC(NC(=O)OC(C)(C)C)C2)cc(C2CC2)on1.c12nncn1C2 C#Cc1cccc(C(=O)NC2CCCCCN(C(=O)Cc3ncc(Cl)s3)C2)c1F c1(C(N(C2CN(C(C34CC=CC(C3)OC4)=O)C2)C)=O)ccc2c(c1)CC2 Cc1cn2c(C(=O)NC(C)C(CO)NC(c3cc(C(N)=O)c[nH]3)=O)c(Cl)nc2s1 N1(C(C2(SCC)CC2)=O)CCC2(CC1)CC(NC(C1CC(O)(C#N)C1)=O)CCO2 Cn1cnc2c(NCC3CNC(=O)O3)nc(N3CCC(SC(F)F)C3)nc12 N1(C(CCSCC(C)C)=O)CCC(C)N(C(c2ccsn2)=O)CC1 C1(O)(CC(N2CC3CC(O)C3C2)C(=O)NC)CCN(C(=O)OC(C)(C)C)CC1 c1(C(=O)NC(C)CCCNC(C2CCC3CC2CO3)=O)cc2cc(Cl)cnc2[nH]1 N1(CC(C)(C)OCC#C)CCCC(N(CC)CC)C1 C=C(C)CC(C(=O)N1CCC(C(=O)NCCCc2ncn(C)n2)(CO)C1)OC C(C(CC(C)C)C(=O)NCC(=O)OC1CC1)NC(C(CCC)OCC)=O C1(NC(C2(C)CCNC(=O)C2)=O)C2CCC1CN(C(C1CCC3CC13)=O)C2 C1(NC(C2CCC(C3CC3)CC2)=O)CCOC2(CCN(c3nnc(O)s3)CC2)C1 C(=O)(C(O)CCC(C)C)N(CCOC)CCNC(=O)Cc1sccc1C C(C(C)(C)C(=O)NC1CCC(CCNC(c2cc(OC(F)F)n(C)n2)=O)C1)SC C(c1ccc(S(C)(=O)=O)o1)=CC(=O)NC1C(CNC(c2ccc(OC)cn2)=O)C1 Cc1c(C(=O)NC2CCCC2CNC(=O)CC2CC2)cc(C)c2ncccc12 CC(C)C(CNC(=O)COC1CCOC1)NC(C1(C(C)C)COC1)=O c1(C(C)C)nccc(=NC2CC(NC(C3CCC(=O)N(C)C3)=O)C2)[nH]1 C1(C)(C(N2C3C(CNC(CS(CC)=O)=O)C(C3)C2)=O)CC(C2CC2)=NO1 C#CCCC(O)C(=O)N1CCCC(N(C)C(c2csc(C)c2)=O)C1 C1(F)(CNC(C(CO)N(C)C)=O)CCC(CNC(c2ccc(=O)oc2)=O)C1 N1(C(c2nccc(CC)c2)=O)C2CCC1C(CNC(C1CC3(CCO1)CC3)=O)C2 C1(CC)C(C(=O)N(C2CCC(NC(=O)CSc3nncs3)CC2)C)CCN1C c1(N(C)Cc2ccco2)nc(=NCC2(CO)CC3C=CC2C3)[nH]c2c1CCC2 N1(C(c2cc(C)cc(Cl)c2)=O)Cc2ccccc2CC1C(=O)NC(C)C1CC1 CC#CCCCC(=O)N1CC(O)(CN(c2cnn(C)n2)Cc2ccccc2)C1 c1(OCC)ccc2c(c1)OCC(C(=O)N1CC(F)(F)C1C1CC1)=C2 c1(-n2cc(CCCC(C)O)nn2)cccc(C(=O)NCCCOCC2CC2)c1 C1(C#N)(OC)CC(C(=O)NC(c2nc(C(=O)N(C)CC3CCC3)co2)C)C1 CC1CC(=O)NC(C(N2CC3CC2CN3C(C2(C(=O)N(C)C)CC2)=O)=O)C1 C1(O)(C(N2CCC(C(CNC(C(C)SC(C)C)=O)(C)C)CC2)=O)CCCCCC1 C1(NC(c2cnc(C)nc2O)=O)CCN(C(=O)CCC(F)F)CCC1CO N1(C(c2ccc(CNC(c3coc(CO)c3)=O)s2)=O)CCCCC(CO)C1 c1(C(N2CCC(NC(c3c(OC)nccc3)=O)(CF)C2)=O)ccc(O)cc1Cl C12(C(N3CC(C(N(C4CCN(C(C)=O)CC4)CC)=O)OCC3)=O)CCCC1CCC2 N1(C(C(N2C(c3nc(C)on3)CCC2)=O)=O)CC2(C)C(=O)NC(=O)C2(C)C1 N1(C(c2c(C)sc(Br)n2)=O)CC2CC(NC(=O)CCCC3CC3)C1C2 Cc1scc(C(=O)NCC2CCCN2C(=O)C(C2CC2)N(C)C)c1C1CC1 C(=O)(C(CC(C)C)N(C)C)N(CCCNC(=O)CS(=O)CC)CC C1(CCC)CCCCN1c1nnc(CCCP(C)(C)=O)n1CC1CCOC1 C1(C(=O)NC2(CCC=C)CC2)CCCN(C(=O)C(C2CCCCC2)F)C1 C1(C(CO)NC(C(C)CC2CCC2)=O)CCN(C(=O)CCc2cnoc2)CC1 C1(C(=O)NC(CC=C)CNC(c2nonc2N)=O)CC2(CCO1)CC2 CC1CN(c2ccc(F)cn2)CCN1C(=O)NCc1ccc(Br)cn1 N1(CC(=O)N(CC(=O)NCCC(=O)OC)C)C(C)CCC1C Cc1ccnc2c(C(N3CC4(CCC4NC(c4cncc(Cl)c4)=O)C3)=O)cnn12 C(C(C)(O)CC(=O)NCc1nnc(C(F)F)o1)OC c1(CN2C(C(=O)NCCNC(C)=O)CC3(CC3)C2)cc(Cl)c(Cl)cc1C c1(CC(=O)NC(c2cccc(Cl)c2)CNC(C(CC)OC)=O)cc(Cl)n(C)n1 Cc1ccc(C=CC(N2CC=CC2(C)C(=O)NCC(C)(C)OC(C)C)=O)cc1 C1(CNC(Cc2nc(C)[nH]n2)=O)CN(C(=O)CCN2CCCC2)CCC1(C)C N1(C(C2CCCC(O)C2)=O)CCC(COC2CCN(Cc3c(C)ocn3)C2)CC1 c1(C(=O)Nc2nc(-c3c(C)cnc(F)c3)sc2)cccc2cn(C)nc12 n1(CC)cc(Br)cc1C(=O)N(C)CC1CCCCN1C(=O)COC(C)C C1(C(=O)NCC(CN(C)C(c2ccccc2NC(N)=O)=O)(C)C)CN2CCC1C2 N=c1nc(C(c2csc(Cl)c2)NC(N2CCC2C2CCCC2)=O)cc[nH]1 C12(CC(N3CCCN(C(C4C(C)C4)=O)CC3)=O)CC3CC(CC(C3)C1)C2 CCC(C)CC(C(=O)N1CCC(C(=O)N(C)C)C1)NC(=O)Cc1ccns1 Cc1cnc(NCCCC#N)c(S(=O)(=O)NCCc2cnns2)c1 C(=O)(CN=c1cc[nH]cc1)N1CCC(NC(COCCC=C)=O)(CC)CC1 C1(NC(C=C(CCC)CCC)=O)COC2(CCN(C(C3CCS3(=O)=O)=O)CC2)C1 c1(CC(=O)N(C2CCCC(NC(CCSC)=O)C2)C)ccccc1S(C)(=O)=O CC(C(=O)NCCCC1(NC(=O)CC2(C)CC2)CC1)C(=O)N1CCOCC1 c1(CC(C)NC(N2C(C)CSCCC2)=O)cc(F)c(F)cc1F N1(C(C(COC)COC)=O)CC2(CNC(=O)C(c3ccccc3)O)CCC1C2 Cc1nc(C(=O)NC(C(=O)NCC2CCCCCC2)C2(C)CC2)sc1C c1(C(=O)NC2CC(C)N(C(=O)CC#N)C2)cc2n(n1)CCNS2(=O)=O C(=O)(C(C)(C)CC(C)C)N1CCC(N(C(=O)Cc2ccccc2CO)CC)C1 C1(CNC(C2CC(=O)N(C3CC3)C2)=O)C2CN(C(c3sc(Br)cc3F)=O)CC12 C1(NC(c2c(CC)c[nH]c2)=O)COCCC1C(=O)NN1CCC1C(N)=O C(C(F)(F)C(=O)N1CCC(C(C)CNC(c2ncccc2F)=O)CC1)OC Cc1nnc2n1CCCC2C(=O)NC(C)(CNC(=O)CCCN(C)C)C1CCC1 C(C1=C(C#N)CCC1)N1C(CC(CC)Sc2ccccc2)CCC1 CC1C(NC(c2cc(O)n(C)n2)=O)CC2CCC1N2C(C1(S(N)(=O)=O)CC1)=O c1(CC(=O)NC2CCCC(NC(C=NOC)=O)C2)ccc2ccoc2c1 CC1(C(=O)NC2CC(CNC(C3CC3c3ccncc3)=O)C2)CCC(=O)N1 N1(C(CN(C(C(C)C)=O)C)=O)Cc2cccc(CNC(C3CCOC(C)C3)=O)c2C1 c1(CCC(N2CC3C(NC(c4c(C)ccs4)=O)(C3)C2)=O)ccccc1C#N c1(OC)cccc(C(N2CCCC2CC2CC2)C(=O)NN(C)CC2CC2)c1Cl C1(NC(CCCCC(C)C)=O)CCN(C(c2nccc(C#N)n2)=O)C12CCCC2 C1(NC(C(C)=C(C)C)=O)CC(C(=O)NC2CCC3(CC3)C2)C12CCC2 C12(C(NNC(c3c(N)cc(O)cc3)=O)=O)CCCC(C1)C(=O)NC2 N1(c2n(CC=C)c(-c3c4c(nn3C)CCCC4)nn2)CCc2nccc(N)c2C1 c1(CSCC(=O)NC2(C(=O)NCCOCC)CC2)[nH]c(-c2ccccc2)cc1C N#Cc1ccc(C(N2CCC(OCCNC(C34C=CC(CC3)C4)=O)CC2)=O)cc1 Cc1cc(=NC(=O)C(=O)NCC(C)NC(c2ccn(C)c2C)=O)[nH]o1 C(=O)(CS(=O)(=O)C1CCCC1)NCC1CN(C(C(CC=CC)C)=O)CC1(C)C c1(C(=O)O)c(F)cc(CN2CCCC(C(=O)NCC3CCOC3)C2)cc1F N(C1CCC(NCc2cccc(O)c2Cl)c2ccccc21)C(=O)OC(C)(C)C c1(CC)ccc(N(C(=O)CC2C3CN(C(=O)C(n4ccc(C)n4)C)CC23)C)cc1 N1(C(C(C)N(C(C)=O)C)=O)CCC2CCN(C(=O)CC(C)F)CC12 c1(C(N2CCC3(NC(C=COCC)=O)C(CC2)C3)=O)coc2c1CS(=O)(=O)C2 N1(C(CN2CC(CC)C2)=O)CCC(NC(=O)CCc2cncs2)C(O)C1 C(C(=O)N1CC(CNC(c2n[nH]c(C)n2)=O)C1)(C(C)C)OCC c1(-c2cc(CNC(N(C3CCSCC3)C)=O)no2)ccc2c(c1)OCCO2 c1(CC)ncccc1C(=O)NC(CC(=O)NCCC1CCCCO1)C1CC1 c1(CC)nc(C)oc1C(=O)NC12CC(NC(=O)Cc3ccc(C(=O)OC)s3)(C1)C2 C(=O)(C(C)C(C)(C)C)NCC(C1CCN(C(C(C(=O)OC)OC)=O)CC1)C C(C(=O)NC(C)CCN(C)C(c1ccc[nH]1)=O)(SC)SC C1(=CC(=O)NC2CN(C(C3(O)CCC3)=O)CCC2CO)C2CC3CC(C2)CC1C3 C(=O)(CC(C)N(C(=O)C(C1CCOCC1)O)C)NCCOCC(=O)OC Cc1cccnc1CCC(=O)NC1CN(C(C2CC3(CCC3)C2)=O)CC1F CC(F)CC(=O)NCC(C)N(C)C(c1cnc(CNC(=O)OC(C)(C)C)o1)=O C1(CC)(CNc2cc(Nc3cnc(C(F)F)s3)ncn2)CCCN(C(C)(C)C)C1 N1(C(c2c(OC)csc2)=O)CC2CN(C(=O)Cc3ccc(Br)c(OC)c3)CC12 Cn1cc(C(=O)NC23CC2CN(C(C2CCC(CC(F)(F)F)CC2)=O)C3)nc1O C12(CNC(C(C)OCCCC)=O)CN(C(c3c(C)ncn3O)=O)CC1CCO2 C1(SC)CN(C(=O)NC(C)C(F)(F)C(F)(F)F)C2(CCCC2)C1 N(C(=NCC(C)C)NCc1cccc(Cl)c1C)C(C#C)C(C)(C)OC C(CC(C)(C)C)(c1n(CC(=C)C)nnn1)NCCc1nc(CC)cs1 c1(C(N(C2CCC(NC(COCCC)=O)C2)C)=O)cnc(O)c([N+](=O)[O-])c1 c1(CC)cc(O)ccc1NC(N1CC(O)(c2nn[nH]n2)C1)=O c1(OC)c(C(=O)Nc2ccc(-n3cnnn3)cc2C)sc(C)c1Br c1(C(=O)NC(CNC(C2CCC(=O)N2)=O)C2CC2)cncc(C(F)(F)F)n1 c1(COC)oncc1C(=O)NCC(O)CNC(c1ccc(C(C)=O)[nH]1)=O CCC(CCC(=O)NC(CC(N)=O)c1cn(CCC(C)O)nn1)OC N1(C(C#CC(C)(C)C)=O)CC2CC1CN(C(C1CC3CCC1C3)=O)C2 c1(NC(C)C(=O)NC2(C)CC(C(=O)O)CS2)ccc(C(F)(F)F)cc1 N1(C(c2ccc(CCC)s2)=O)CC2C3CCC(C2C1)N(CCOC)C3 C1(CNC(c2ccc(O)cn2)=O)CCCCN(C(=O)Cc2ccccc2Br)C1 CCCCC(F)C(=O)N1CC(C(=O)NC(c2cscn2)C)(SC)C1 c1(C(=O)NCC(CNC(c2nc(C(C)C)oc2)=O)O)cncc(F)c1 c1(C(N2CCC2(C)C(=O)NC)C(=O)NCC=C)cc(C(C)C)nn1C CCC(C(=O)NCCNC(c1csc(CC(F)F)n1)=O)C(F)(F)F N1(C(=O)COCCc2ccncc2)CC2CC(C1)CN(C(c1ccoc1)=O)C2 N1(Cc2cn(CC(CC(C)C)n3cc(CO)nn3)nn2)CCCCCCC1CO c1(C(N(CCSC)CC)=O)ccc(NC(=O)C(C2CCCO2)OC(F)F)cc1 Cc1ncccc1CC(=O)NC(CC1CCCC1)C(=O)NC1CC(Cl)(Cl)C1 C12(C(=O)NC(C)Cc3nncn3C)C(NC(c3ccn(CO)n3)=O)C3CC1C2C3 C1(CC)CNC(=O)CN1C(c1cc([N+](=O)[O-])c[nH]1)C(=O)NCSc1ccccc1 CS(=O)(=O)C1CC(C(N2CC3(CCC3NC(c3cccnc3)=O)C2)=O)C1 C1(NC(=O)NC(CCN2CCCCC2)C(=O)O)CCCC2(CC1)CC2 O=C1CCCC(C(=O)NC(CO)C(=O)NCc2nncs2)CC1 C#Cc1cccc(CCNC(=O)N(C2CCN(C3CCC3)C2=O)C)c1 C(CCCC(=O)NC(CCC1CC1)C(=O)NCc1cc(O)ccc1C)(OC)OC CC(C)C(C)(O)C(=O)NCCCC(c1ccccc1)NC(=O)CNCC(C)(C)C c1(C2CN(C(=O)CCc3ncco3)C2)c[nH]c2ccc(F)cc12 C1(CNC(=O)CCc2ncc(F)cn2)CCCC12CCN(C(=O)CC1CC1)CC2 c1(CCC(N2C(C)CC(CNC(c3cc(Br)n[nH]3)=O)C2)=O)nc2cccnc2[nH]1 N1(C(C2C3CN(C(C(c4ccccc4)=O)=O)CC32)=O)CCC12CCCCC2 CC(C)(C)C#CC(=O)NCC1CC(F)(CNC(=O)C(C)(C)c2ccccn2)C1 C1(CC(=O)N(CCCN(C)C)C)C2CCCC2N1C(c1ccc(O)cc1F)=O c1(OC)c(SCCCC(N2CCN(C(=O)C(F)CC(C)C)CC2)=O)c(=O)c1=O c1(CC)cc(C(=O)NC2CCCC2NC(=O)C=Cc2cncc(O)c2)c(C)nn1 N1(C(C2N(CC)CC2)=O)CCN(C(=O)C#CC(C)(C)C)C(c2ccccc2)C1 C1(NC2CCN(C(CC)C(F)F)C2)CCC12CCC2 c1(C(=O)NCC(=O)NC(C)CC2CCC2)ccnc(O)c1 C1(C(=O)NC23CC(NC(c4ccccc4F)=O)(C2)C3)CCC(C2CC2)C1 c1(C(N2CC(C(C)NC(=O)CCc3nc[nH]n3)OCC2)=O)ccc(S(C)=O)cc1 C1(NC(C(CC=C)C)=O)CC(C)CN(C(=O)CN(C)C(c2ccsc2)=O)C1 CCCCC(CCC)NC(C1CCC2(CC2)N1C(c1cnn(C2CC2)c1)=O)=O CC(C(=O)NCCOCCNC(=O)CCc1ccc[nH]1)C(C)c1ccccc1Cl c1(C(C)OC)nc(C(=O)NCCCCCNC(=O)C(F)=CC2CC2)co1 Brc1nc2c(s1)CN(c1cc3cc[nH]c3cn1)CC2 C(=O)(C(C)(C)Cc1cnn[nH]1)NCCCN(C(=O)C(C)CCN(C)C)CC c1(-c2cn(-c3cccc(SC)c3)nn2)nccc(SC)c1F c1(OC)c(Br)ccc(C(N2CCC(OC(C)C)CC2)C(=O)NC(C)C)c1F Cc1nccnc1C(=O)NC1CCCCC1CNC(C1CC(NS(C)(=O)=O)C1)=O N1(C(CNCCCC(C)C)=O)CCN(C(=O)OC(C)(C)C)C(CS(C)(=O)=O)C1 c1(-c2cn(CCCCCCNC(C3C(OC)C3)=O)nn2)cc(C)cc(Br)c1 C(C(=O)NCC1(CO)CCN(C(C2CSC2)=O)C1)(C(C)(C)C)OC CCCCC(F)C(=O)NCCNC(=O)CO.C1CCOCCOCCO1 C1(NC(C(C2(C)CC2)NC(=O)CCn2ccnn2)=O)CCOC1=O C1(CNC(c2cc(CC)oc2C)=O)CN(C)CCN1C(=O)Cn1cnnn1 C(C(=O)NCCCN(C(=O)CCCc1ccc(OC(F)F)cc1)C)(C(C)C)SC N1(C(c2c(NC(C)C)cccn2)=O)CCCC(NC(=O)CSC2CC2)C(F)C1 Cc1cc(C(=O)N(CCC(C)NC(=O)CCc2ncco2)C)c(C(F)(F)F)o1 c1(CNC(c2c(C)nc(O)[nH]2)=O)nnc2n1CCN(C(C1CCCN1N=O)=O)C2 CC(C)CC(C(=O)NCC12CC(NC(c3cncc(F)c3)=O)(C1)C2)C(N)=O CC1(C)CN(C(c2cc(C(F)F)[nH]n2)=O)CC1C(=O)NCC1(C)CCCS1 Cc1ccc2oc(-n3cc(CCC4CCC4)nn3)cc2c1 CC1(C)CN(C(=O)COC2CCC(F)(F)CC2)CC1CNC(C1CC(CF)C1)=O C1(C(C)O)CCCN(C(=O)CC2CN(C(C3(CO)CCC3)=O)CCO2)C1 c1(C(=O)NC2C(NC(c3cnc(C)[nH]3)=O)CCC2)cc2occ(Br)c2[nH]1 c1(NC(C2C(NC(CNC(C=C)=O)=O)CCC2)=O)cc(Cl)cc2ncoc12 c1(C(=O)NC(C(=O)OCCNC(=O)OC)C)ccccc1C N1(C(c2cc(C)oc2)=O)CCC2(CCC2)C(NC(c2cnc3scc(C)n23)=O)C1 c1(CC)cc(NC(=O)NCC(C)CC2CC2)c(C)cc1F CCC(CCCC(=O)NCC(C)(C)C(C)O)NC(c1nccnc1C)=O c1(C(=O)NC(C(CO)NC(CC=CCC)=O)C)cnc(O)c2cncn12 C1(C(=O)NCC(C(=O)OCC)C)CN(C(C2CCCC2O)=O)CC1(F)F C12(NC(c3ccc(C(C)C)cn3)=O)COC(C1)C(NC(C1CC1C(F)(F)F)=O)C2 C1(CNC(C(COC)(F)F)=O)CCN(C(=O)C(=O)NC2CC2)CC1(F)F c1(CN2CCC3(C(C(=O)Nc4cc(OC)nnc4)C3)C2)cnc2ccccn12 c1(NC(C(=O)NC(CC(=O)OCC)C)=O)ccc(F)c(I)c1F C1(N2CCCC(C(N(C)Cc3nccn3C)=O)C2)CCCCC1S(C)(=O)=O CC(C)C(c1cn[nH]c1)NC(CC1(CNC(=O)C(C)c2cncs2)CC1)=O CC1(O)CC(C(=O)NC2CC(NC(=O)CCCc3ccncc3)C2)C1 Cc1cc(C)c(NC(=O)CCCN(C)C(c2nnc(S)n2C)=O)cc1C N1(C(C(CCCCC)O)=O)CCOC2(CCCN(C(=O)Cn3cncc3C)C2)C1 c1(C(=O)NCC2(F)CC(CNC(CC(C)SC)=O)C2)cc2ncccn2n1 N1(C(C2C(C)(Br)C2)=O)CCC2(COC(CNC(=O)CN3CCCCS3(=O)=O)C2)C1 C(=O)(C(C)=NOCC#N)NC1(CC(=O)N(C(C#C)C)C)CC1 C1(C(=O)NC(c2scc(C)n2)C)C=CCN(C(c2ccnc(CO)c2)=O)C1 C(=O)(C1=C(SC)CCCC1)NCC1N(C(c2cccc(COC)c2C)=O)CCC1 N1(C(C(C)NC(CC)(C)C)=O)CCC(C2CC2)C1C(=O)NC1CCC(O)C1O C(=O)(CCCC(F)(F)F)NC(C1CCCN(C(c2cnc(SC)n2C)=O)C1)C C(CCCC(=O)NCC(CC1CC1)C(=O)NCCCc1cccs1)(OC)OC CC1CCc2c(sc3nc(CNS(=O)(=O)c4ccccc4Br)nc(O)c23)C1 C(N=c1nc2[nH]ncc2c[nH]1)c1c(NC(C(CC)NC(C)=O)=O)c[nH]n1 c1(CNC2(c3onc(C)n3)CCCC2)ccc(-c2nn[nH]n2)cc1S(C)(=O)=O N1(C(c2c(CC(C)C)onc2)=O)CCN(C(=O)CC(=O)NCC2CC2)CC1CF N1(C(C(C)OCC)=O)CCCC1(C)CNC(=O)CCCc1cnn[nH]1 CN1CC2(CCN(C(C3CCN(C(=O)Cc4ccc(Cl)cc4)C3)=O)CC2)C1 c1(C2C(NCc3cn(CC(N)=O)nn3)C2)cccc(Cl)c1Cl C(CO)(CC(C)(C)C)NC(C1N(C(c2c(C)occ2)=O)CC(O)C1)=O C1(CNC(C2CC3CCC(C2)C3)=O)CCCC12CCN(C(C1SCCS1)=O)CC2 N1(C(CC(CC=C)NC(CC=C)=O)=O)CCCC2OCCC2C1 C1(CC(=O)O)(C(=O)Cn2cc(-c3ccc(C(F)(F)F)cc3)nn2)CCCCC1 CC(C(=O)NC1COCCN(C(c2ccc(CO)s2)=O)C1)S(C)(=O)=O N1(C(CN2CCCCC(=O)C2)=O)CCC(C2CC2)C1C(=O)N(CC1CC1)CC1CC1 c1(C(C)NC(c2cc(CNC(=O)CCc3ccc[nH]3)[nH]n2)=O)ccc(O)nc1 Cc1cc(O)ccc1CNc1ncc(-c2ccnn2C(C)C)cc1O CCCC(CC)CC(=O)NCC(C)(C)OCCNC(c1scnc1Cl)=O N(C(=NCCF)N1CCCC2(C1)CC2(F)F)CC(C1CCC1)OC Cc1ccccc1C(C)C(N1CCCC1CNC(=O)CCc1cccc(O)n1)=O N1(C(C(=O)N(CC2C(C)CN(C3CC3)C2)C2CC2)=O)CCOCCC1C1CC1 C1(C(N2CCCC(CCC#C)C2)=O)CN(C(=O)CC(C)F)CC1(F)F N1(C(C2(C)ON=C(C)C2)=O)CCC2(CC1)OCCCC2NC(c1cccnc1)=O c1(C(=O)NCCC(C)NC(c2ccn(C3CCC3)n2)=O)ccc(CC(C)(C)O)s1 c1(NC(C2CN(c3ncc4[nH]ncc4n3)C2)=O)cccc2c1CN(c1nccs1)C2 N1(C(c2[nH]cc(CC)c2)=O)CCc2nc(CNC(c3cccnc3C)=O)sc2C1 N1(C(CSCCC)=O)CCC(NC(=O)COc2cccc(C(C)C)c2)C1(C)C c1(C(N2CCC3(CC(NC(C4(CO)CCCO4)=O)C3)C2)=O)c(F)ccc(F)c1F CC1CC(C(=O)NCC(=C2CN(C(=O)CCC3CC(C)(C)CO3)C2)F)CCS1 C(=O)(CCC(F)F)N(CCCNC(CC1N(CC)CCC1)=O)C N1(C(C2C3C(=O)C4C(C3)C42)=O)CC2(C(=O)N(CCCO)CCO)CCC1CC2 CCC(C)C(O)CC(=O)N1CC(O)(CN(C(=O)C=Cc2cccc(F)c2Cl)C)C1 CCC(CCCC(=O)NCC1CC(O)C12CCC2)NC(C1C2CCC(F)C12)=O c1(C(=O)NCCc2cc(C(N(CC(C)O)CCO)=O)no2)c[nH]c2cnccc12 c1(C(N2CCCC(C)(NC(CCCCOCC)=O)C2)=O)ccc([N+](=O)[O-])c(C)c1 c1(CC)ccc(CNC(=O)C(C)(C2CCC2)NC(=O)CCCN(C)C)cc1 N1(C(CCCCOCCC=C)=O)CCC(C)C(NC(c2cn(C)nc2CC)=O)C1 C#Cc1cnc(C(N2CC(O)(C(C)NC(C34CCOC(C)(C3)C4)=O)C2)=O)c(C)c1 c1(CNC(=NC)N(C)NC(CCC)COC)cc(Cl)ccc1OC C12(C(N(C3CCC3)CCN(C)C)=O)CC1CN(C(c1cc[nH]n1)=O)C2 N1(C(c2c(C)c[nH]n2)=O)CCCC(O)(CNC(=O)CCOC2CC2)C1 c1(C(N2CCC(CC(=O)Nc3c(OC)ncnc3)C2)=O)cc(F)c(F)cc1Cl CC1CCC(CO)N1C(C1CCN1C(C1CCC(=O)N1C)=O)=O CC(Cc1nccn1C)N=c1[nH]c(=NC2CCc3ncsc3C2)c2sccc2[nH]1 C1(CNC(C2(C)CCOCC2)=O)CC2(CC2)CN1C(=O)Cc1c(O)ncnc1O c1(C(=O)NCCN(C(C2(O)CCC(C)CC2)=O)C)cnc2ncnn2c1C(C)C CC1Cc2ccc(Br)cc2CN1.C1(C=O)CSC2(c3ccccc3)CCC(=O)N12 c1(OC)ccc(C)nc1C(N1CCCC1CCNC(C1CCCOC1C)=O)=O C1(C)(NC(C(CC)N(C)C(c2ccccc2C#N)=O)=O)C(C)(C)C1(C)C C(C1=CCN(C(=O)CCc2ccsc2Cl)CC1)NC(c1nc(CC)oc1)=O c1(C(N2CCCC(N(c3c(C)cnc(Cl)n3)CCO)C2)=O)cc2ncccc2s1 C1(CNC(=O)Cc2ccns2)CC(NC(c2cc(F)cc(F)c2)=O)C12CCC2 c1(-c2cn(C(C(=O)N(C)CC3(CO)CCC3)C)nn2)ccc(Cl)nc1 N1(C(C(CC)=CC)=O)CCN(C(=O)Cc2ccc(O)cc2)CC1CC c1(C2(CNC(c3n(CC=C)nnn3)c3ncc(C)s3)CCC2)cc(Cl)ccc1Cl c1(CC(=O)N(C)CC2(O)CN(C(CN(CC(C)(C)C)C)=O)C2)cccc(F)c1 Cc1cnc(F)c(C(C)NCC2CCN2C)c1 C1(C(=O)NCCN(C)C(C2(C(N)=O)CCC2)=O)CCOC1C(F)(F)F c1(C(C)C)cnn(C)c1C(=O)NCCC1COCCN1C(=O)C(CCO)N(C)C N1(C(C(CCC)O)=O)CCC2(COC(CNC(C3CCCN(C(C)=O)C3)=O)C2)C1 C(=O)(CC(C)(F)F)NC(C)CCN(C(=O)CCc1ccn(C)n1)C c1(OC)cc(C#N)ccc1S(=O)(=O)Nc1ccc(-c2cnn(C)c2)s1 C1(NC(CCNC(=O)C=CCl)=O)CCN(C(c2cccc(N3CCCC3)c2)=O)C1C C1(NC(CN(C(C)=O)C)=O)C2CC1N(C(c1cncc(CO)c1)=O)C2C N1(C(Cc2n(C)nc(C(F)(F)F)c2)=O)CCC2CCC(NC(=O)CC(=O)N)C1C2 c1(CC(C(=O)NCC2(O)CCN(C(c3c[nH]c(=N)s3)=O)C2)O)c(F)cccc1Cl CCCC(C(=O)N1CCC(NC(=O)C(C2CCS(=O)(=O)CC2)O)CC1)S(N)(=O)=O c1(NC(C2N(C(c3cc(CC)ncc3)=O)CC2)=O)ccc2[nH]nc(Cl)c2c1 CC1N(C(c2c(CNC(C3(C)C=CCCC3)=O)cnn2C)=O)CCCC1(C)C C1(C(=O)NCC2C(CNC(C3CC(SC)C3)=O)C2(C)C)(CO)CCCO1 C1(NC(C2(OC)CC(CO)C2)=O)CC2(C1)CC2C(N1CC(N2CCNC2=O)C1)=O N1(C(=O)NC)CCCC(C(=O)NCC(CC)NC(C2(NC(C)=O)CCCC2)=O)C1 C1(CNC(=O)CCC2CC2)C=CCN1C(c1nocc1Cl)=O C1(C(=O)NC(C2CCN(C(C=Cc3c(C)n[nH]c3)=O)CC2)C)CC(=O)NC(C)C1 CC1CN(C(=O)CCn2cnnn2)CCC1NC(c1cc(Cl)cnc1O)=O C=C(Cl)C(C)(C)C(=O)NCC1CCCN(C(=O)C(F)CC2CCCCC2)CC1 Cc1nc2[nH]c(COC(=O)C=Cc3ccc(O)c(OC(C)C)c3)cc2s1 Cc1cc(C(=O)NCC2(C)CCN(C(=O)CN3CCCC3C)C2)nc(O)n1 c1(C(N2C(CC(=O)NS(=O)(=O)CCCl)COCC2)=O)c(Br)cc(F)c(F)c1F C(=O)(C#CC1CCOCC1)N(C(N1CC(C(C(=O)O)C(C)(C)C)C1)=O)C1CC1 c1(CC(=O)N(CCN(c2c(C(=O)OCC)cccn2)C)CC)c(C)nn(C)c1Cl C#CCC(CC#C)C(=O)NC1CCN(C(c2nc(Cl)ccc2N)=O)C1 c1(C(=O)NC(CC(C)Nc2ncnc(Cl)c2CO)C)cccn2cnnc12 c1(NC(c2nc(NC(c3c(C)scc3)=O)sc2)=O)ccccc1[N+](=O)[O-] C1(CC=C)(NC(c2ncccc2Cl)=O)CCN(C(C2CC2F)=O)C1 CC1C(NC(=O)C=Cc2ccc(F)cc2)C(C)CCN1C(C1OCC1(C)C)=O Cc1cc(O)cc(=O)n1CC(=O)NCC1CCN(C(c2cc3occc3[nH]2)=O)C1 c1(CNC(C=CC(C)NC(c2cccnc2S)=O)=O)ccnc(F)c1F N1(C(COC2(C)CCC2)=O)CCC(c2cccc(F)c2)C(NC(C2CCC2)=O)C1 N1(c2c(C(=O)OC)cnc(Cl)n2)CC2CCC1C(NC(=O)CC1CCC(C)C1)C2 c1(NC(c2cc(C)c(Br)cc2)=O)ccc2c(c1)CCN(C(=O)C(C)(C)F)C2 C1(C)(CCNC(c2c(CC)nn[nH]2)=O)CCN(C(=O)C(CC2CC2)OC)CC1 c1(C(=O)NC2CCC(CCNC(CC3CC(OCC)C3)=O)C2)cc(C)cc(C)n1 N1(C(c2cc(OC)c(C)cc2)=O)CC2(CCC(CNC(C3(CCF)CC3)=O)O2)C1 C1(CNC(c2ncc(NC)nc2)=O)CCCCN(C(=O)C(C)C(C)C)C1 c1(CNC(C(=O)N(C2CC2)CC)(C)C)c(C)n[nH]c1C C(=O)(C#CC1CCOC1)N1CC(C(C)NC(=O)CCOC2CCCC2)C1 c1(OC)cc(C)cnc1C(=O)NCCCN(C)C(C1CCO1)=O c1(C(N2CCC(N(C(C(C)NC(CC)=O)=O)C)CC2)=O)c(F)ccc(C)c1Cl N1(C(COC(CC)C)=O)CCN(C(=O)C(O)Cc2cnc[nH]2)CC1CO C1(NC(CCCC#C)=O)CCC(C)(C)CC1CNC(=O)C(CO)N(C)C c1(C(=O)NCC=CCNC(CCCCC)=O)ccc2c(O)nc(=O)n(C)c2n1 CC(C)C(C#N)C(=O)N1CC(C(N2CC3(CC(O)C3)C2)=O)CC1(C)C c1(C(=O)NCCC(C)NC(c2csc(C3CCCO3)n2)=O)c[nH]c(=N)s1 c1(OC)ccc(C(=O)NCC(C)(C)CCNC(=O)CC2CCC(OC)C2)cc1Cl CC(C)C(CO)CCNC(C1CC=CCC1NC(=O)C1=CCCCC1)=O C1(CC(=O)N(CC(F)Cl)C)CC(C)(C)CN1C(=O)CCc1ccn(C)c1 Cc1cccn2ncc(C(=O)NCC3CC(NC(C4(C)CC4(F)Cl)=O)C3)c12 c1(CC)cccc(CC(=O)N(CC(C)N(C)C(C2CC3CC3C2)=O)C)c1 Cc1cc(F)ccc1NC(C1(CNC(=O)OC(C)(C)C)CCCCCC1)=O N1(C(=O)CC=Cc2ccccc2)CCC(C2CC2)C1CNC(C12CC(CO1)C2)=O C(C)(CC(=O)NC1CC2CC1N(C(c1cnc(N)c(Cl)c1)=O)C2)(C(F)F)N(C)C c1(OC)n[nH]c(C(=O)N(C)CC2CCCCN2C(=O)CC2C(=O)ON=C2C)c1Cl c1(C(=O)NC(c2nc(COC)on2)C)c(Cl)ccc(Br)c1Cl c1(CC=C)cccc(C(N2CCCC(CNC(c3cc(OC)cnn3)=O)C2)=O)c1 N1(C(CN(C(C)C(C)C)CC)=O)CC(CCN2CCCC2)C1 C12(NC(=O)Cc3cncc(O)c3)CCCC1CN(C(=O)C=CSc1nc[nH]n1)C2 c1(N2CCC(C)CC2)nc(N2CCc3cccnc3C2)c2c(n1)CCC2 C1(CNC(COc2ccc(C)cc2)=O)CC12CCN(C(C1CC(O)C1)=O)CC2 O=C(C(=O)NC1CSCSC1)NCCOCC1CCC1 CCC(C)C(=O)C(=O)N(C)CC=CC(=O)NCCC1(C)CCCO1 C1(C#N)(C(=O)NCCCN(C)C(C2CCC(CC(F)(F)F)CC2)=O)CCCO1 N1(C(CCOCC#C)=O)CCC(F)C(NC(=O)C(C)C(C)(F)F)C1 C1(C(=O)NCC2CC(NC(c3cc(CCC)oc3C)=O)C2)CCCC1S(C)(=O)=O Cc1ccc(C(=O)NC2CCC(NC(c3nnc(Cl)cc3N)=O)CC2)c(O)n1 CC(O)C(C(=O)NCc1nn[nH]n1)NC(=O)C=CCF Cc1c(NC(C)C)cccc1NC(=O)NC1C2CC2CN1C(=O)CC1CC(F)C1 C12(C(=O)NCC3N(C(C(C)CO)=O)C4C(C3)COC4)CC3CC(C1)CC(C)(C3)C2 c1(N(C)C)cc(Br)ccc1CN=c1[nH]c(CC(=O)Nc2ncc(Cl)cc2O)cs1 C=C1CCC(C(=O)NC23CC(NC(=O)C(C)Sc4ccc(F)cc4)(C2)C3)CC1 N1(CCNC(c2c(COC)scc2)=O)CCN(C(=O)CCNC(N)=O)CC1 N1(C(c2n(C)nc(Cl)c2)=O)CCC2(CNC(=O)CC3CCC(=O)NC3)CCCC12 CCCCC(O)C(C)C(=O)N1CC(=O)CC1C(N1C2COCC1C2)=O c1(C(=O)NCC(CNC(C2(C(C)C)CC2)=O)F)cccc(-c2cnco2)c1 N1(C(c2cc(OCC)no2)=O)CC2CC(NC(C3(C)CC3(F)F)=O)C(C2)C1 C1(C(=O)NCCC2N(C(CSCC)=O)CCSC2)Cc2ccc(C)cc2S1 C(=O)(CC(C)(C)OC)NCC(=O)NCC(=O)N(C1CCC(C)C1)CC C1(CC(=O)NOCc2cn(C3CSC3O)nn2)(N(C)C)CCOCC1 Cc1cn2nc(C(=O)NC3CCN(C(=O)CCOC(C)C)CC3F)cc(C)c2n1 C1(C(N2CCC(C)(CNC(c3c(C)scn3)=O)CC2)=O)C2CCC3C(C2)CC13 c1(C(N2CC3C(CC(=O)NCC(COC)OC)C3C2)=O)nccc2[nH]ccc12 c1(C(N(CC(C)SC)C)=O)cc(O)nc2c1CN(C(=O)CCC1CCOC1)CC2 C(=O)(CC(CN(C)C)CC)N(CC(CNC(CC1(COC)CC1)=O)C)C C1(NC(c2ccc(C#C)c(C)c2)=O)CC2CCC(C1F)N2C(C12CSCC1C2)=O Cc1cc(C(N2CCN(C)CC2CNC(C2(C(F)(F)F)CC2)=O)=O)nc(O)c1 CC(CCNC(=O)C=Cc1cncs1)CCNC(=O)CC(c1cccc(F)c1)C C1(NC(CCCC2C(C)C2)=O)C2CC3C(C2)C13C(=O)NCC1CC(N(C)C)C1 Cc1cnc(C(=O)NCC2CCN(c3ccnc(C4CCC4)n3)CC2C)cc1Cl c1(C(N2CCC3(C(NC(=O)CCc4cncs4)C3)C2)=O)cc2c([nH]1)CCCC2 N1(C(=O)CC2CCC2)CCC(C(=O)NC(CO)CCF)C1 N1(C(C(=O)NC(C)(C)C)CC2(C#N)CC2)CCOCC1CC1CCCO1 CCC(CC)C(F)C(=O)N(CC(N1CC(O)(CC(C)C)C1)=O)C1CCC1 N1(C(C(c2cnn(C)c2)C)=O)CC(NC(=O)CC(F)(F)Br)C2(CC2)C1 C1(C(N2CCC(OC3CCC3)CC2)=O)CSCCN1c1ncncc1F C(=O)(C1CCC(=O)c2cccn21)NC1C(NC(=O)CC2(O)CCCCCC2)CC1 c1(C(N2CCC(NC(CC=CC=C)=O)C(CO)C2)=O)ccc(S(C)(=O)=O)[nH]1 CC1(C)CC(CNC(Cc2cc(CO)no2)=O)CN(C(=O)CCN2CCC2)C1 C#CCCCC(=O)NCC1CCC(C(=O)NC(C2CCOCC2)C)O1 C1(C)(C(=O)NC(C2CCN(C(C3(C)CC(F)C3)=O)CC2)C)COC(=O)OC1 C1(CC(=O)NCC(C)CNC(=O)CC2CC(C(F)F)C2)CCCN1C c1(C(=O)NCC2CN(C(C(Cc3c(C)n[nH]c3C)C)=O)C2)cccc([N+](=O)[O-])c1 c1(C(=O)NCCC(C)N(C(c2cc(C)c(F)cc2)=O)C)ccc2ncc(C)n2c1 CC(c1ccco1)=CC(=O)NCCC1CCN(C(=O)CNc2cccnc2)C1 C1(CC)C(NC(=O)Cc2ccc(Cl)cc2)CCCN1C(C1COCC(C)(C)O1)=O N1(C(c2csnn2)=O)CCCC2(CCN(C(c3cc([N+](=O)[O-])ccc3O)=O)C2)C1 N1(C(Cc2ccc(OC)cc2C)=O)CCC2(C1)CN(C(=O)C(C)O)CC(C)O2 C1(CNC(c2cc(SC)c(C)o2)=O)CCCN(C(C2CCCC(C)(C)O2)=O)CC1 c1(SC)nc(=NC2CCCC2C(=O)Nc2cc(C(F)(F)F)no2)c(C#N)c[nH]1 N1(C(c2ncc(OC(C)C)nc2)=O)CCOC2(CCN(C(=O)C(C)(C)C)CC2)C1 c1(OC)cc(N)c(F)cc1C(N1CCC(NC(C2CCCCO2)=O)C1C)=O n1(CCOC)ncc(C(N2CCOC(CCNC(=O)C(C)=C3CC3)C2)=O)c1C CCC(C(=O)NC(C)(C)CC(N1CCNC(=O)C1C)=O)C(C)(C)CC C(C(C)C)(C(F)(F)F)NC(COC1CC(NC(C(COC)C)=O)C1)=O C1(CCC)(NC(C2CC(Cl)(Cl)C2)=O)CCCN(C(C2CC3CCC3C2)=O)C1 C1(CC(=O)NC2(CNC(c3ncn(C)n3)=O)CCOC2)CCCC2(CC2)C1 Cc1ccc(C(N)=O)cc1C(=O)NCC1(NC(=O)C(C)(C)c2ccccc2)CC1 C(=O)(C1=C(COC)N(c2ccc(F)c(Cl)c2)C(=S)NC1c1cncn1C)OCC c1(C(=O)OCCOCOC)ccc(C(=O)N(C)CCO)[nH]1.C12(CCC1)C(=O)NC2 N1(C(CSCCC)=O)CCC(O)C(N(C(=O)COC(C)(C)C)C)C1 C(=O)(CC(C)CC(C)C)NC1CCC(NC(c2cc(C(C)=O)on2)=O)CC1 CC1CN(C(=O)C(=Cc2cscn2)F)CCN1C(=O)C(C)C(=O)OC(C)(C)C c1(C(C(=O)NC(CNC(c2cccc(CC)n2)=O)(C)CO)C)ccc(F)c(F)c1 C1(CNC(=O)COC2CC2)C=CCN1C(C1CCCN1C1CC1)=O C(=O)(C(C)S(N)(=O)=O)NCCC(=C)CNC(=O)C=CC1CCCN1C C(=O)(C1=CC(O)CCC1)NCC(CC=C)NC(=O)C=Cc1ccco1 C(=O)(C(O)CCNC(=O)Cc1cccnc1)NC(C=C)(C)CC S(=O)(=O)(c1ccc([N+](=O)[O-])c(C)c1)NCC(C(=O)OC)Cc1cccc(C)c1 c1(C(=O)NCC(CCCC)NC(=O)C=CSC)cc(CCC)nc(O)c1 C(=O)(C1=NN(CC)C(=O)CC1)NC(CC)CN(C(=O)C(C)=CC(C)(C)C)CC C1(NC(c2nc[nH]n2)=O)CCOC1C(=O)NC1COCC1O N1(C(C2ON=C(C)C2C)=O)CC2CN(C(c3conc3C)=O)CCC12 C(=O)(C(C)(C)C(C)C)N1CCC(N(C(c2c(CCC)[nH]cc2)=O)CCO)C1 c1(CSC)ccc(C=CCNC(=O)NCC2(C3CCC3)OCCO2)cc1 N#Cc1nnn2c1CCC(C(=O)NNC(=S)Nc1cccc(Br)c1)C2 N1(C(c2c(C)scn2)=O)CCC2CC(NC(C3CC4CCC3C4)=O)CCC2C1 C(=O)(C1=CS(=O)(=O)CCC1)NCCC(C(C)C)NC(c1cc(OC)nc(Cl)c1)=O N1(C(c2ccc(COC)cc2)=O)CCCC(O)(CNC(=O)Cc2ccsc2C)C1 C(=O)(CS(=O)CCC(F)(F)F)N1CC(O)(C(C)NC(c2c(C)coc2C)=O)C1 Cc1nn(C)c(C)c1C(N1CCCC1(C)CC(N1CCC(c2cc[nH]n2)C1)=O)=O Cc1cc(F)ccc1-c1cn(CCN(C(=O)CC2CCC(C#N)C2)C)nn1 CCC(C)CC(C)N(C(=O)C(O)C1CN(C(C2CCC(=O)O2)=O)C1)C C12(NC(c3cc(SC)c(C)o3)=O)CCN(C(c3cnco3)=O)CCC1C2 C1(NC(CCC(=O)NC)=O)CN(C(=O)C(F)(F)Cc2ccccc2)CC(C)(C)C1 C1(NC(c2cnc(C)nc2)=O)CCN(C(c2cnn(C)c2)=O)CC12CCC2 C1(NC(CN(C2CCC2)C)=O)CCC12CN(C(C1(C)C=CCC1)=O)C2 Cc1c(C(=O)NC2(CN(C(=O)CC(C)NC(N)=O)C)CC2)sc2nccn12 CCCC(O)C(=O)N(C(CNC(C1(C)CC1Br)=O)C1CC1)C C(=O)(C(C)(C)CCOC)N1CC(COC(C(CC=C)C)=O)C(OC)C1 C1(CNC(=O)C(F)CC2CC2)(CO)CCN(C(c2ccc(F)c(Cl)c2)=O)CC1 c1(C(C)C#N)cccc(N(C(=O)Oc2nn[nH]n2)Cc2ccccc2)c1 C1(C(=O)NC(C(C)NC(c2cc(CC(C)C)[nH]n2)=O)(C)C)CC2CCC(C1)C2O CCCCC(C)C(=O)NCCC(C)CCNC(c1cn(C)nc1COC)=O c1(C(=O)NC(Cc2ccc(OC)cc2)C(=O)O)cnc2c(c1)CCS(=O)(=O)C2 c1(N(CCCN(C)C2CC2)C(=O)CC2CCCCC2O)ccc([N+](=O)[O-])c(C#N)c1 c1(C(=O)NCC(C)N(C(=O)CC(c2cccc(F)c2)C)C)cc2n(n1)CCCN2 C(=O)(CCC(C)C#N)N(C)CC1N(C(Cn2c(C)csc2=O)=O)CC(F)C1 c1(C(=O)NCCN(C(COCCCC)=O)C)cc(O)nc(C)n1 N1(c2nnc(C(C)C)o2)CCCC2(CN(C(=O)C(C)CF)CCO2)C1 C1(CNC(CCCc2nc(C)sc2)=O)CCCN(C(c2cncc(F)n2)=O)CC1 Cc1ccc(OCC(=O)NCC2C=CC(NC(C3(C)COC3)=O)C2)c(C)c1 C=CCCC(C)(C)C(=O)N1CC2=C(C1)CN(C(=O)Cn1ncccc1=O)C2 c1(NC(CC2CCN(C(COCCC#C)=O)C2)=O)cccc2nn[nH]c12 Cc1ccc(O)cc1C(N1CC(F)(F)CC1CCNC(C1(C)CC1C)=O)=O c1(C(=O)NCC2N(C(c3ccc(SC)o3)=O)CC=C2)nnn2c1CSCC2 C1(CNC(C(C)SC)=O)CCCC(NC(c2ccn(C3CC3)c2C)=O)C1 C(=O)(C(CC(C)C)NC(=O)C(c1sc(C(F)(F)F)cc1C)N(C)CC1CC1)OC N1(C(c2c(COC)cccc2)=O)CC2CCN(C(c3coc(Cl)n3)=O)C(C2)C1 c1(C(=O)NCC2CCN(C(=O)COC3CC3)C2)c[nH]c2ccncc12 N1(C(c2cc(COC)sc2)=O)CC2(CC2)CC1CNC(=O)C(C)C(F)(F)F CC(C)C(CCN(C)C(C1CC1(Cl)Cl)=O)NC(C1(CC(C)=O)CCCC1)=O Cc1cc(N)c(F)c(C(=O)NC(c2ccccc2)C2CCCCC2)c1F C#Cc1ccc(C(=O)NC(C)CCCCNC(C2C3CCC(F)(F)C23)=O)cc1F Cc1c(C(=O)NCC23CCC(C2)N(C(=O)C(C)N(C)C)C3)[nH]c2ccccc12 Cc1cc(CC(=O)NCC2(O)CCN(C(=O)CSCc3ncc[nH]3)C2)cc(C)c1 C1(CCCC(=O)NCCC(=C)CNC(c2cnc(Cl)c(Cl)c2)=O)CCCC(=O)N1 CCCCC(CC(=O)NC(c1cccnc1O)C)NC(=O)Cn1cncn1 C1(CNC(C2C(C)CCO2)=O)CN(C(=O)CCCCN(C)C)CC(C)(C)O1 C#Cc1cccc(C(N2CCCCC2C(C)NC(=O)C(F)CCC(C)C)=O)c1F O=C(C1=CNC2=NCCC2=C1)NC12CC1CN(C(C1CCCC3(CCC3)O1)=O)C2 C=C1CCN(C(=O)C=Cc2cncn2C)C(C(=O)NCC2(SCC)CC2)C1 NC1(CNC(c2oc(-c3ccccc3)nc2-c2ccccc2)=O)CC2CCCC12 N1(C(c2cnc(CC)[nH]2)=O)CCC2(CC1)CCN(C(C1(n3cnnn3)CC1)=O)C2 C(C1=NOC2COCC12)NC(C(CC(F)F)NC(C1CC2CCC1CC2)=O)=O N1(C(C2(CC#C)CC2)=O)CCN(C(=O)CN(C2CCSC2)C)C(CCO)C1 c1(OC)ccc(Cl)c(C(=O)NCC(CC(C)C)NC(C2COCCC2(F)F)=O)n1 c1(C(N2CCCC(CNC(CCC=CC)=O)CC2)=O)ccc2c(c1)C(=O)CCS2 CC1CC2(CCN(C(=O)C(C)(F)C(C)(C)F)CC2)CN1C(=O)CCCCCC#N C1(NC(C=C(C)CNC(=O)C(O)C(F)(F)F)=O)(CO)CC2CCCC12 C(=O)(C(C)CC(=O)OC)N1CCC(C(=O)NC(c2cn(CC)nc2)C)C1 C=Cn1nncc1C(=O)NC1CCCCC1CNC(=O)COC N1(C(CC(COC)(C)O)=O)CCC(F)(F)C(CNC(=O)CN(C(=O)C(C)C)C)C1 c1(-n2cc(CN3CCC(NC(C#CC(C)C)=O)CC3)nn2)c(F)cccc1F c1(C(N(CCCNC(C(CC)Oc2ccccc2)=O)C)=O)nn(C)cc1C(C)=O C(CCC(=O)NC1CC1)N(CC(O)C(N)=O)C(CC1(C)CC1)=O c1(C(N2C(C)CCC(CNC(CCC(=O)OC)=O)C2)=O)cnc(O)n(C)c1=O C1(C(=O)NC2CCC(NC(C3(C(F)F)CC3(F)F)=O)CC2)CC2(C1)CC2(F)F CCC(CCC(=O)N(CCCN(C)C(C)=O)C)NC(c1ccc(Cl)c(N)c1)=O C=CC(C)CC(=O)NC1C=CCCC1C(=O)NCc1ccsc1 Cc1nc(O)sc1C(=O)NCC(C1CCN(C(=O)C=Cc2cnccn2)CC1)C c1(C(=O)NCC(C(=O)N(CCSC)CC)C)cnc(O)n1CC CN1CC(C(=O)NC(C2CCCCC2)C(=O)Nc2cncc(F)c2)NC1=O c1(OC)c[nH]c(C(=O)N(C(C)CNC(c2c[nH]cc(Br)c2=N)=O)C)cc1=O c1(N(C)C)cccc(C(N(Cc2coc(NC)c2)Cc2ccccc2)=O)c1 c1(C(NOCCC(C)=O)=O)cnc(C)nc1-c1ccco1 c1(C(N2C(CNC(C(=O)NC(C)C)=O)CC(O)C2)=O)cnc(C2CCC2)nc1O Cc1ccc(OCC(=O)N(CC(C)NC(=O)Cc2cc(Cl)cnc2C)C)c(C)c1 c1(CN2CCC(CC(=O)NC(C)C#N)C2)cccc(C2CC2)c1Cl c1(C(N2CC(CNC(c3c(=N)cc[nH]c3)=O)OCC2)=O)cc(Cl)cc(F)c1F N1(C(C(COC)OC)=O)CC2CCC1CN2C(=O)CN1C(=O)C(=O)N(C)C1=O c1(CC(C)C)cccc(CO)c1.c12nc(-c3ccc(C(C)(C)C)cc3)nn1C2 C(=O)(CC(C)(C)C(C)(F)F)N1CC(O)(C(C)NC(C2CC2(C)C)=O)C1 N(C1CCOc2cc(F)cc(F)c21)C(N1CCn2ncc(Br)c2C1)=O C(=O)(CCC(F)(F)F)N(CC(=O)C(=O)OC(C)(C)C)C.c1(C(CC)N)nn[nH]n1 C1(C(=O)NCC2(C#N)CCCC2)CCN(C(c2n[nH]c(=N)[nH]2)=O)CCO1 N1(C(CC(=O)N(C)C)=O)CC2CC(CNC(C3COCCC3(F)F)=O)C2C1 c1(C(=O)OC)cc2cn1C(C1CC1)n1c(nnn1)CO2.C1(SC)CC1 C(=O)(C1=CCCCCC1)NCC1C(C)CN(C(c2ccc(OC(F)F)nc2)=O)C1 CN1CC(NC(=O)C(CNC(c2ccc(C3CC3)o2)=O)CC2CC2)CC1(C)C c1(C(N2CCCC(n3cc(CNC)nn3)CC2)=O)ccnc(S(N)(=O)=O)c1 c1(CCC(=O)NCC(CC)NC(=O)C=CCN(C)CC)csc(=N)[nH]1 c1(C(C(=O)N(C2CN(C(=O)C(F)OC(F)(F)F)C2)C)(C)C)ccccc1Br c1(CC)[nH]nc(Cl)c1C(=O)NC1CC(CNC(C2COC(C)(C)C2)=O)C1 CCC(O)CC(=O)NCc1ncoc1C1CN(C(=O)CCc2ncc[nH]2)C1 c1(C(=O)NC(C(N2C(CC)CCC2)=O)CC)cccc2[nH]ncc12 N1(C(C(C)CS(C)(=O)=O)=O)CCC2CCN(C(c3ccnn3C)=O)CC2C1 C12(NC(C=CSC)=O)COC(CNC(c3cc(Cl)cs3)=O)(C1)C2 Oc1ccc2c(c1)C1(CCN(Cc3scnc3C(F)F)CC1)CN2 CC(C)CC(CNC(=O)CC1CCNC(=O)C1)NC(c1cnc(CC2CC2)s1)=O CC1c2cc(F)cc(F)c2CCN1C(N1CCCC(CNC(=O)OC(C)(C)C)C1)=O c1(-c2cccc(NC(c3cc(C(C)=O)[nH]n3)=O)n2)cccc2c[nH]nc12 c1(C(N(CC(C)N(C(=O)CCCCN2CCCCC2)C)C)=O)cc2sccc2s1 c1(C(=O)NC2(CCNC(CC(C)C3CCCO3)=O)CC2)csc(C#N)c1 C#CCCCCC(=O)NCCN(C(=O)C(c1cnn(C)c1C(F)(F)F)C)C N1(CCC(C)(C)NC(C(CC)NC(N)=O)=O)CCN(C(c2ccc(C)s2)=O)CC1 C1(CC(=O)NCc2cc(C)cs2)(NC(CCCOC(C)=O)=O)CCCCC1 CN1CCCC1C(N1CCC1C(=O)NOCC(O)CO)=O c1(C(=O)NC2C(CNC(=O)CSc3ccccc3)CC2)ccc2nncn2c1 C1(O)(CCNC(CC2(C=C)CC2)=O)CCCN(C(=O)CS(=O)(=O)NC(C)(C)C)C1 C1(CNC(=O)C(O)c2cnc[nH]2)CC2CCC1N(C(c1nc(F)ccc1Cl)=O)C2 N1(C(Cn2ncc(C)c2)=O)CCC2(COC(CNC(=O)CCCN(C)C)C2)C1 Cc1nc(O)ccc1C(=O)NC1CCCN(C(=O)CC2CC=CCC2)C1C Cc1ccc(C(N2CC3(CCCN3C(c3ccc(O)c(I)c3)=O)C2)=O)c(C)c1Br N#CC1(NC(c2cc(Br)cnc2Br)=O)CCN(C(c2cc(F)nc(F)c2)=O)C1 CC1CN(C(=O)C(C)(O)C2CC2)CC1C(=O)NC(C)C(O)C(F)F c1(OC)ncc(Cl)c(=NC2CC(CNC(=O)Cc3cc(F)ccc3F)C2)[nH]1 C1(CCNC(C(C(C)C)F)=O)CCN(C(C23CCC(CC2)CC3)=O)CC1(F)F C1(NC(C2CC(C(F)(F)F)C2)=O)CCN(C(=O)Cc2cnc(C3CC3)[nH]2)CC1O C1(C(=O)NC(CNC(CCOCC#C)=O)(C)C)Cc2ccccc2C1C C1(NC(C2CC(C)(C)C2)=O)CN(C(C2(Cl)CC2)=O)CC1O C12(C(=O)NCCC(C)NC(=O)CC3CCCN(C)C3)CC3CC1C2C3 C(CN=c1nc(N2CCC(C3CC3)C2)c2cnn(C(C)(C)C)c2[nH]1)OC(CC)C C(=O)(CCCC(=O)NC(CO)C(C)NC(c1ccc(C(C)C)cn1)=O)NCCC CCCCC(CNC(=O)CCCN1CCCC1)NC(=O)CCc1nc(C)c(C)[nH]1 c1(C(CC)C)ccccc1OCC(=O)NCCC(C)NC(C1CC=C(C)CC1)=O Brc1c[nH]nc1C(c1nnnn1CCCC1CC1)NCCCC1CCCCC1 N1(C(CCC2(NC(c3nc(CC)oc3)=O)CCCC2)=O)CC(F)CC(F)C1 CC1CN(C(c2coc(CO)c2)=O)CC(C)N(C(=O)C(c2ccncc2)C)C1 CCCC(CCC)CC(=O)N1CC(CO)CC1C(=O)Nc1ccc(OCOC)cc1 N1(C(CNC(CCC)=O)=O)CCC(CNC(=O)CN(C)C(=O)OC)CC1C c1(C(N2CC3C(N(C(C(C)OCCCCCC)=O)C)C3C2)=O)cnc(N)c(Cl)c1 c1(NCC(C(C)C)OC)nc(N(C)CCc2ncc(C)s2)nc2c1ncn2C Cc1cc(Br)ccc1CN1CCCC1C(=O)NCCCCCO c1(NC(CC(CC)NC(C2CC(COC)C2)=O)=O)cnc(C)c(C)c1 c1(C(C)(C)NC(c2ccn(C3CCOCC3)n2)=O)ccc(Cl)cc1 Cc1cc([N+](=O)[O-])cc(C(N2CCC(NC(=O)C3=C(C#N)CCC3)CC2)=O)c1Cl c1(CC)nn(C)c(Cl)c1C(N1CCC(NC(c2ccccc2)=O)C(CO)C1)=O C(C(C(C)(C)C)NC(C1(C)CCSCC1)=O)NC(c1c(CC)scc1)=O N1(C(CCCn2c(C)ncc2)=O)CC2CN(C(c3ccc(C(F)(F)F)[nH]3)=O)CC12 C(=O)(C(CC(C)C)ONC(c1nn(C)cc1C)=O)N(CCN(C(C)=O)C)C CC(C(=O)NC1CN(C(c2ccc(C(F)F)c(F)c2)=O)CC2CC12)C(F)(F)F N1(C(c2snc(C)c2Br)=O)CC2ON=C(CNC(C3(C)CC3)=O)C2C1 C(=O)(C1=CCOCC1)N(C)CC1N(C(C(C(=O)OC(C)(C)C)OC)=O)CCOC1 CCC(C)N=c1cc(NCC2COC(=O)N2)nc(C(F)(F)F)[nH]1 C#Cc1cnn(CC(=O)NCCN(C(c2cccnc2-n2nccn2)=O)CC)c1 N1(C(C(C)OCC(C)C)=O)CCC(C)(C)C1CC(=O)NCCS(C)(=N)=O CC1CCNCCC1N(CC(C)CCl)C(c1c(F)cncc1F)=O N1(C(C(C#C)(C)C)=O)CCC2(CCC2NC(c2ccc(CCC)c(N)c2)=O)CC1 CCCCCCCCC1C(=O)N1CCOC.C(C(Cl)Cl)N.CCCOC N1(C(C(CC)=CC)=O)CC(CNC(=O)C(O)C2CCC2)C(C)(C)C1 C1(NC(CNC(=O)OC)=O)CC2CCC1(CNC(C1CC(S(C)(=O)=O)C1)=O)C2 N1(C(CCC(C)OCC)=O)CCC2CN(C(=O)CCOCC(F)F)CCC12 CC1CNCCC1NC(=O)C(=O)NCC(C)(C)c1cccs1 C(C(C(=O)OC)C(C)C)(c1n(CCCOC)nnn1)NCCCc1nc(C)no1 N1(C(c2oc(CC)c(C)c2)=O)CC2CCN(C(c3ccc(Cl)cc3O)=O)C2C1 C1(CNC(C2CCCN(C(C)C)C2)=O)CCN(C(=O)C(F)C2CCC2)CC1C c1(C(N2CCC3(NC(CSCCCC)=O)C(CC2)C3)=O)nc2nccc(C)n2n1 N1(CC)CCOC(C(=O)N(CC(C)(C)CNC(C2(C)CC(C)=NO2)=O)CC)C1 C1(NC(CN(CC)CC)=O)CCN(CCNC(=O)COCCOC)C1 CC(CS(C)=O)C(=O)NCCCCNC(c1ccc(-c2cnc[nH]2)cc1)=O C1(C(C)NC(CC2ON=C(C)C2)=O)(NC(C2CCN2C(C)C)=O)CCOCC1 C1(C(=O)OC)CCCN(C(=O)C(=O)Nc2cc(C)c(O)c(C)c2)CC1F C1(OCC(=O)N(CCCN(C(C(C)NCC)=O)C)C)CCC(C)CC1 N1(C(CCCCC(=O)OC)=O)CC2C3CCC(C2C1)N(Cc1ccccc1)C3 C(C1=NOC2CCCCC12)NC(N1CC2C3COCC3C2C1)=O N1(C(=O)CC2=CCCC2)CCC2(CCCCC2NC(=O)C(F)(F)C(F)F)CC1 C(CCCCCNC(C1(C)COCCO1)=O)NC(C(C)(C)n1cc(Cl)cn1)=O C(=O)(C(O)(C(C)C)C(F)(F)F)OCc1c(C)cc([N+](=O)[O-])cc1 c1(C(N2CC(=C(CNC(c3ccn(CC)n3)=O)F)C2)=O)ccc(O)c(N=[N+]=[N-])c1 C(=O)(C(C)S(=O)(=O)C(C)C)NC1CC(F)(CNC(C=CCN(CC)CC)=O)C1 C1(SC)CN(C(c2cccc(C3CCCOC3)c2)=O)CC1NC(=O)CCF CCC(CC(=O)N1CCC(C)(C)C(CNC(=O)C(F)(F)C2CCCC2)C1)C(F)F N1(c2c(C(N)=O)cnc(Cl)n2)CCCC2(NC(C3CCOC3)=O)CC2C1 C(=O)(C(C)CS(C)(=O)=O)N1CC(CNC(c2nncc(C)c2)=O)N(C)CC1 c1(C(C)C(=O)NCCC2CCCN2C)ccc2c(c1)OCO2 c1(OC)cc(C(=O)NC2CC(NC(c3cc(C)c[nH]3)=O)C2)c2ncccc2c1 Cc1cc(O)c(C(C)C)cc1C(=O)N(C1CN(C(C2CC=CCO2)=O)C1)C C1(N(C(=O)Cn2cccn2)C)CN(C(C2C3COCC23)=O)CCC1O C1(CNC(C2CC3(C2)CC(CO)C3)=O)CCCC2CN(C(C3(O)CCC3)=O)CC12 c1(C(=O)NCCC(C)N(C(C(CCC)=CCC)=O)C)cnc(O)cc1C(F)(F)F c1(OC)ccc(C(O)C(=O)N(CCCCNC(c2nc(O)sc2C)=O)C)cc1 c1(C(=O)NCc2cccc(NC(CCOCCC)=O)c2)nsc2c(Cl)cccc12 Cn1cc2c(n1)CCN(C(C1CCCC1NCc1cccc(I)c1O)=O)C2 C1(C(=O)NCC2(OC)CCN(C(=O)C(C)SC(C)C)C2)OCC2CCCCC12 CCCCC(F)(F)C(=O)NCCc1n[nH]cc1C(=O)NC1CC12CCC2 Cc1cc(C(N2CCN(C(c3cnc(O)s3)=O)CC2CO)=O)c2n[nH]cc2c1 C1(C(N2CCC(C(C)OCC)CC2)=O)CN(C(C2(SC)CC(=O)C2)=O)CCN1C C#Cc1ccc(NC(=O)CCCC(C)(C)NC(c2ccnn2C)=O)c(C)c1 c1(OC(C(N2CCCC(NC(c3ccn(C)n3)=O)C2)=O)(C)C)ccc(F)c(F)c1 C1(CNC(CC2(OC)CCC2)=O)CN(C(C2CCOC(C)(C)C2)=O)CCC1(C)C C1(C2N(C(CCCOCC)=O)CCC2)CCN(C(c2ncnn2C(C)C)=O)CC1 c1(SCC(=O)N(C2CCN(C(COC(CC)(C)C)=O)CC2)C)ccc(C#N)cc1 C(=O)(C(C(=O)NCCN(C(=O)C(O)CC1CCOCC1)CC1CC1)C1CC1)OC c1(OC)c(F)ccc(F)c1C(=O)Nc1cnc2n1CCOC2 C1(CC(=O)NCCN2CCC(O)CC2)CCCN(C(=O)CN2CCCC2)CC1 C(=O)(CCC(=O)NC(CC(=O)NC(CN(C)C)CO)C1CC1)NC c1(C(N2C(C)(C(=O)NCC(C)SC)CCC2)=O)cc(C)c(F)cn1 c1(C(N(CCn2cc(-c3cccc(F)c3)nn2)CC)=O)sc2cccnc2c1Br CC(C)CC(F)(F)C(=O)NCCC1CCN(C(c2ccc(OCCF)cc2)=O)C1 Cc1cccc(C(N2CC3CC2C3C(=O)Nc2cc(Cl)ccn2)=O)n1 C1(OC)(CNC(N2CC(=O)N3CCC3C2)=O)CC(C)CC(C)C1 C1(NC(c2c(C(C)(C)C)[nH]cn2)=O)CC12CCN(C(=O)C(F)C(C)(C)O)CC2 C(=O)(CCCCCCCOC(C)C(=O)NC(C)=O)OCC.C12CCN1C(=O)C2 Cc1cc(C(=O)NCCNC(=O)CC2CCCC(C)(C)O2)c2ccccc2n1 c1(C(CC)C)ccc(C(=O)NCC(O)CN(C(=O)C#CC(=O)N(C)C)C)c(O)n1 CC1(CCCCNC(=O)NCc2cccnc2S)NC(=O)NC1=O C=C=C(C)CC(=O)NCCC1CSCCN1C(=O)CN1CCCCC1 C(C1c2ccccc2CCN1C(C1CC(=O)N(O)C1)=O)NC(c1cscn1)=O C1(NC(C2(COC)CCCC2)=O)CCN(C(C2CC2(C)C)=O)C1c1ccccc1 C(c1ccncc1)=CC(=O)NC(CC(C)NC(C1(n2cccn2)CCCC1)=O)C c1(C(N(C2CN(C(c3ccc(NC)cc3)=O)C2)C)=O)ccc(S(=O)(=O)CF)nc1 N1(C(c2cc(C)nn2C)=O)CCC2(CCCC2NC(c2cccnc2S)=O)C1 n1(CC)cnc2c(NC3CC(CC#N)C3)[nH]c(=NCc3cnccn3)nc12 C1(NC(C(c2ccc(F)cc2)C)=O)CCC12CN(C(=O)C=Cc1ccsc1)C2 C(CN=c1cc(C)nc(C2CCC2)[nH]1)N(C(CC(CC)C(C)C)=O)CC N1(C(C2(C#C)CCCC2)=O)CC(CNC(c2ccc3c(c2)CC3)=O)C(C)(C)C1 C1(CNC(C(C)S(N)(=O)=O)=O)(NC(C2C3CCCOC23)=O)CC2CCC1CC2 N1(C(C2(C)CCCN(C)C2)=O)CC2CC(C1)CN(C(C1CCCOC1)=O)C2 C1(C(=O)NCC2N(C)CCN(C(C3CC3C3CC3)=O)C2)CN2CCCN1CC2 N(C1CCCc2nn(C)cc21)c1c(C)c(N2CC(C(N)=O)OC(C)C2)ncn1 c1(CCC(N2CC(N(C(CC(C(=O)OC)C)=O)C)C2)=O)cncc2ccccc12 C1(CNC(=O)CSC(F)F)CCC2(CCN(C(C3CC34CCOCC4)=O)CC2)O1 N1(C(CC(=O)OC)=O)CCC2(CC1)CC(C(=O)Nc1cccc(O)c1Br)CO2 N#CC1CN(Cc2cncs2)CC1NC(c1cnc(Cl)s1)=O N1(C(c2cc(CCCCC)[nH]n2)=O)CCC(C)C(NC(c2n[nH]c(C)n2)=O)C1 c1(C(=O)NC2C(C)CCN(C(C3(F)CC3)=O)C2)nn(C)cc1S(N)(=O)=O NC(=O)CC(C(=O)N1CCC(c2ccc(C3CC3)nc2)C1)N1CCCCC1 N1(C(c2ccc(C(N)=O)nc2)=O)CC2CC(NC(=O)CC3CCSCC3)C1C2 C1(CC(=O)N(C)CC2(O)CN(C(c3cc(CC)n(C)n3)=O)C2)NC(=O)CNC1=O C=CCC(C)(CC)C(=O)NCC(C)(C)CC(=O)NCc1cc(C)ccn1 CC(F)(F)C(C)(C)C(=O)NC1CCC2CCN(C(c3cncc(Cl)c3)=O)C12 c1(C(=O)NCC2(F)CCN(C(COC3(C)CCC3)=O)C2)scc2c1CCCC2 c1(OC)ccc(C(N2CCC(O)(C(C)NC(C3CC(C)(F)C3)=O)CC2)=O)c(F)c1 Cc1n[nH]c(C)c1SCC(=O)N(C1CCCN(C(C2(C)CCCN2C)=O)C1)CC c1(C(=O)NC2CCCC(CNC(C3C(OC)CC3)=O)C2)ccc(OC)nc1C c1(C(=O)NC2C3CCN(C(c4ccc(C=C)cc4)=O)C32)ccc2nc(Cl)nn2c1 N1(CC(=O)NCC(C)N(C)C(c2ccc(C3CC3)o2)=O)CCOCC1=O N12CC3(C1)CN(CCO3)C(=O)OCCCC2=O.C(CC)(C=O)=CCCC N1(C(=O)CO)CCC2(CC1)CCN(C(C1CCC3C(C1)C3(F)F)=O)C2 C(CC(C)(C)CNC(C1CCCCO1)=O)NC(C(C)Cc1cnc[nH]1)=O C1(c2c(OCC(NOCC)=O)c[nH]n2)CC(C)CCN1C(=O)C(C)C(=O)OC S(=O)(=O)(c1ccc(NC2CCC(P(C)(C)=O)C2)c(F)c1)N(C)Cc1sccc1Cl S(=O)(=O)(c1ccc2c(c1)CCCNC2)N1CC(CS(C)=O)C1 c1(C(=O)NC(CCC)C(=O)N(C(C)CCO)C)ccc2[nH]ccc2n1 C(=O)(C(C)(C)CCCF)NC(C)CCCNC(=O)COc1ccc(F)nc1 C(CCN=C(NCC1CCC(F)(F)C1)NCC1(NC(=O)NC)CCC1)OCC C=CC1CN(C(C2(Cl)CC2(F)F)=O)CC1NC(c1cn(C)nc1CC)=O C#CCC(CC(F)F)C(=O)N(C1CN(C(=O)C(C)CC2CCCC2)CC1(C)C)C N1(C(COCCCC)=O)CCC(CO)(NC(C2CCN(C)C2)=O)C1 N1(C(C(=O)Nc2cnn(CC)c2C)=O)CC2CCCC(CO)(C1)C2O Cc1cccc2cc(C(=O)NCCOC(C)(C)CNC(=O)Cn3ncnn3)nn12 N1(C(c2ccn(CC)c2C)=O)CCCN(C(=O)C(C(C)O)NC(=O)C2CC2)CC1 c1(C(=O)NC(Cc2n(C)ccn2)C2CC2)cnc(-c2ccc(F)cc2)cn1 S(=O)(=O)(c1cn(C)[nH]c1=N)N(CCO)Cc1cccc(C)c1 C1(CNC(c2ncc(C(F)(F)F)cn2)=O)CC(O)CCN1S(=O)(=O)C1CC1 C1(C(=O)NCCC2C=CCC2)(CC)CCCN(C(C2C3CC4C(C3=O)C24)=O)C1 CC(C)CC(O)CC(=O)N1CCOCC1CNC(c1scnc1C(F)(F)F)=O c1(C(=O)NC23CC(CNC(C(C)SCC)=O)(C2)C3)cnc2cc[nH]c2c1 CCCCC(F)(F)CNC(=O)NCCN1CCC(N=[N+]=[N-])CC1 C(=O)(C#CC(=O)N1CCC(O)(CNC(C2(C(C)(C)C)CCCCC2)=O)C1)N(C)C N1(C(C(C)S(C)(=O)=O)=O)CCC(F)(F)C(CNC(C23CCN(CC2)C3)=O)C1 C1(CNC(c2c(OC)c[nH]n2)=O)CCC(C)N(C(=O)CSCCOC)C1 c1(NCc2cccnc2)ccc(OC(c2cccc(CC)c2)=O)c(Br)c1 C12(C(=O)NC3C(NC(C4(C)CCC4)=O)COC3)CCCN(CC1)C2 c1(C(N2C3C(NC(C(n4ccc(C)n4)C)=O)CC(C3)C2)=O)nn(C)c2c1CCC2 c1(C(=O)NC2CC(NC(CSCCC)=O)C23CCC3)c(C)ccc2c1CCCN2 C(CC(C(=O)N1CC([N+](=O)[O-])C1)NC(=O)COc1ccsc1)OCC N#CCCCC(=O)NCC1CN(C(=O)CC2COCC2O)CC1c1cncn1C C1(NC(C2CCOCC2)=O)CN(C(c2cc(Cl)c(F)cc2O)=O)CCC12CCC2 C#CCCCCCCC(=O)NCC(C)CN(C(=O)C(C)(C(C)C)NC(C)=O)C c1(C(N(C2CCN(C(c3cc[nH]n3)=O)C2)CC)=O)ccc(S(N)(=O)=O)cc1F C(C(=O)NCCCCNC(=O)Cc1nncs1)(C(C)O)NC(C)=O C=CCC(CNC(c1cc(F)cnc1O)=O)C(=O)NCc1cnccc1C c1(C(=O)NC(CC)CN(C(c2[nH]nnc2C2CC2)=O)CC)cncc2[nH]ccc12 CC(C(=O)N(C)CCN(C)C(C1CNC(=O)C(C)(C)C1)=O)C(F)(F)C(F)F c1(NC(N2C(C)(C)CCC2CO)=O)c(Cl)cc(Cl)cc1Cl c1(C(=O)NCCNC(C)=O)cnc2cc(-c3ccc(O)cc3)ccc2c1Cl C(CNC(C1CC(C)N1C(C1(c2ccno2)CC1)=O)=O)(C(F)(F)F)OC C(=O)(C(O)CC(C)C)N1C(CC)CC(F)C1.c12ccc(nc1)C(=O)NC2C1CC1 C=CCC(CC(F)(F)F)C(=O)NCCOc1cccnc1F c1(C(N2CCC(CNC(C3CCCS3)=O)C23CC3)=O)cccc2c1COCC2 Cc1ccncc1CC(=O)NCCCC(C)NC(=O)Cc1ccsn1 C(C(=O)NC1C=CCCC1C(=O)NCCC1(C)CCCO1)(C(C)(C)C)OC N1(C(c2nn(-c3cc(F)cc(F)c3)c3c2CCC3)=O)CCS(=O)C2(CCC2)C1 C1(CNC(c2ncccc2F)=O)CCCN(c2nnc(C(F)(F)F)s2)CC1 N1(C(C2CCN(C(c3nc(C)sc3)=O)C2C)=O)CCCC(C)CC1 c1(C(=O)NCCN(C(c2c(N)cc(Cl)nc2)=O)C2CC2)cncc2c1CCC2 c1(C(C(=O)NCC(C)(O)CNC(C2CC(=C3CC3)C2)=O)(C)O)cccc(F)c1 C12CC(O)CN(C1)OC1C(CC(=O)OC)C(C1)N2.c1(C(=O)OC(C)(C)C)ccco1 c1(C(C2N(CC(C)C)CCC2)(C)C)cc(Cl)cc(Cl)c1.N12CCCC1CNC2=O C12(C(=O)NC3C(C(=O)OC)CC3)CCCC1N(C(=O)CC1COCC(C)O1)CC2 C1(C(=O)NC(C(C)C)C)CCCN(CCNC(C)(C)C)C1 C1(OC)CN(C(C2CC=CC2)=O)C(C)(CNC(c2coc(N(C)C)n2)=O)C1 Cc1cnn2cc(C(N3CC(O)CC3CNC(=O)CCOCC3CC3)=O)cnc12 Cc1nc(C)c(C(=O)NCC2(F)CC(NC(c3ccc(CC(C)C)cc3)=O)C2)s1 C(CC(C(=O)NC12COC(CNC(=O)CCC3CCCC3)(C1)C2)NC(N)=O)SC c1(COC)cnc(OC)c(C(N2CC(NC(=O)CCC3CCOC3)C(O)C2)=O)c1 N1(C(C(CC)OC)=O)CCC(CCNC(c2ncoc2C(F)(F)F)=O)CC1 C1(NC(CC(C)F)=O)CN(C(=O)COCC2CCC2)Cc2ccnn2C1 c1(CC)ncnc(N(C2CCCN(C(C3(C(C)C)COC3)=O)C2)C)c1F C1(OC)CC(CCNC(=O)C=CSC)N(C(C2C(C)(C)C2(F)F)=O)C1 c1(C(C(=O)NCCCCNC(=O)CC2CC=CC2)CO)ccc(Cl)cc1 C1(C#N)(C(N2CC(N(C)C(c3cccc[n+]3[O-])=O)C(O)C2)=O)CCCOC1 C(CNC(=O)C(C)SC)(CC(=O)NCc1nncn1C(C)C)OC Cc1nc(C(N2CC3CC2CN3C(c2cc(CO)ccn2)=O)=O)ccc1F N1(C(C(CC=CC)C)=O)CCN(C(c2cc(C(F)(F)F)ccc2C)=O)C2CCC12 Cc1cc(C(=O)NC2C=CC(CNC(=O)CC(C)C(C)C)C2)c(F)cc1F C(C(C(=O)NOCC1CCCC1)N(C)C)NC(c1c(C)n(C)cn1)=O c1(OC)cccc(OCC(N2CCN(C(C3CSC3)=O)CC2)=O)c1 CCCC(C(=O)NCC1(O)CCN(C(=O)CC2(CO)CCCC2)CC1)S(N)(=O)=O C#Cc1cc(C(=O)Nc2ccccc2C2CCCCC2)ccc1Cl c1(OC)ncc(Cl)c(=NCC2C(C)CCCN2C(=O)CSCc2ccccc2)[nH]1 C1(CCNS(CC)(=O)=O)CCN(C(=O)Nc2ccc(C(C)(C)O)cc2)CC1 N1(C(c2c(C)cnn2C)=O)C2CCC1CC(N(C(=O)CCCCN(C)C)C)C2 C(=O)(C(F)CC(C)C)NC(CN)C(C)(C)C.CC(C)CCCN(C(c1ccccc1)=O)C=O C(C(C)(C)C(=O)N1CCC(O)(CNC(=O)CCOCC2CCCO2)C1)N(C)C N1(C(CC(C)O)=O)CCC2OCCN(C(=O)CCc3ccn(C)n3)C2C1 C1(N(C(CCNC(C)=O)=O)C)CN(C(C23CCCC2(C(N)=O)C3)=O)CCC1O c1(OC(C)C(=O)NC2(C)CC(C(=O)NC(C3C(C)(C)C3(F)F)=O)C2)ccc(Cl)cc1 N1(C(=O)NCC2CCCN2C2CC2)CCc2c(O)ccc(F)c2C1 N1(C(Cc2c(C)occ2)=O)CCCC2(C1)CN(C(C1(C(F)F)CCC1)=O)CCO2 N(C1c2ccccc2CC1NC(=O)C=C1CCC1)C(CC(=C)Br)=O CCC(C)CC(=O)C(=O)N1CCC(C)C(CC(=O)NC2C(=O)OCC2(C)C)C1 C1(C2CCN(c3nc(C4CCCC4)ns3)C2)(NC(c2c(CC)cccc2)=O)CC1 Cc1cc(C(N2CCOCC(NC(c3csc(Br)c3)=O)C2)=O)nc(Cl)c1 c1(C(N(C(C)C(=O)NC(C)CCc2cn[nH]c2)C)=O)ccc(Cl)s1 N1(C(C=Cc2cncc(C)c2)=O)CC(C2CCCN(C(=O)CC(C)C)C2)C1 CC(C(=O)N(C1CN(C(=O)CCc2nccs2)C1)C)C(C)(C)c1ccccc1 C1(NC(CCN(C(=O)CCc2ccoc2)C2CC2)=O)CC2CSCC2C1 C1(O)(C(N(C(C)CNC(=O)CS(=O)CC)CC)=O)CN2CCC1CC2 N1(C(C(C)C2CCCO2)=O)CCCC2(CCN(C(=O)C(F)n3cccn3)CC2)C1 C(=O)(C1=COCCO1)N1CC2C(CNC(C(C)(C)n3cc(Cl)cn3)=O)C2C1 C1(C(=O)OC)CC2(CCS(=O)(=O)CC2)CN1C(=O)C(C)n1cccn1 C1(C(=O)NC2CC(CCC(=O)NCC3CCC4CC34)C2)CCC2(CCC2)O1 c1(C(=O)NCC(C)CC(F)(F)F)n[nH]c2c1CN(C(C1(C)CCOCC1)=O)C2 c1(-n2c(COC(C(C)C)=O)nc(-c3ccccc3Cl)n2)ccc2c(c1)CCO2 N1(C(C2(SC)CC2)=O)CC2CCC1C1CN(C(=O)CCc3ncc[nH]3)CC21 C1(C(=O)OC)(CCNC(=O)NCCCNCS(C)(=O)=O)CCC1 C#CC1CCN(C(c2ccc(CNC(c3cccc(C)c3)=O)cc2)=O)C1 N1(C(c2ncc(CC)cn2)=O)CCN(C(=O)C(O)C(F)(F)F)CC1CCO c1(C(N2CC3C(NC(C(C)NC(=O)NC)=O)C3C2)=O)cc(OC)c(F)c(Br)c1 C(=O)(CC(CC)CCCC)NC(CC=C)CNC(c1cc(CO)oc1C)=O CCCCCCC(C(=O)NC(C)CCCNC(c1ccc(C)nn1)=O)NC(C)=O C1(SC)CCN(C(=O)CCN(CCCO)C(C2(CO)CCCO2)=O)C1 C1(COC)CN(C(=O)C(C)OC)CCN1C(=O)C(O)C1CCCC1 CC(C)CCC(O)C(=O)N1CC=CC(C(N2CCC(N3CC=CC3)C2)=O)C1 C1(C(=O)NC(CCCNC(CSCC(C)C)=O)C)CC(=O)N(C2CC2)C1 N1(C(CCC)C)CC(C(=O)NC(C2CN(c3ncc(C)cn3)C2)C)CC1=O Cc1nc(O)nc(C)c1C(N1CC2CCC2(CNC(C2CC2C2CC2)=O)C1)=O Cn1cc(NC(C2(C)CCN(C(=O)C(C)(C)F)C2)=O)c(C(F)F)n1 C1(C(N(C2CCN(C(c3nccnc3N)=O)C2)C)=O)CC2CC(C1)CC(F)(F)C2 C(=O)(CS(=O)(=O)CCO)N1CCC(CC)(NC(c2csc(C)c2C)=O)CC1 CCC(CC)CCC(=O)N(CCCNC(=O)C(O)CC(F)F)CC C(=O)(C1=NOC2COCC12)NC1(C(=O)NCC(C)SCC)CCCCC1 CC(C)(CC(=O)NCCCCNC(C1CC2CCCN(C1)C2)=O)C(F)(F)F C(CCO)(C(C)(C)C)NC(C=CC(C)NC(c1cc(C)nnc1)=O)=O Nc1ccc(-n2cc(C(=O)NC3CCCOC3)cn2)cc1 C(C(C)C(C)(F)F)NC(C(C1CCCN(C(=O)COC2CCCOC2)C1)C)=O c1(CC)ccc(C(N2CC(NC(=O)CC=C(C)C)C(SC)C2)=O)cc1 CC1CC(NC(c2nscc2Br)=O)CN1C(c1ncccc1Cl)=O c1(CC(=O)NC(c2cn(CC(O)COC)nn2)CCC)ccc(C(=O)OC)cc1 c1(C(N(C2CC3CCCC(C2)N3)c2ncc(C)cn2)=O)nc2ccccc2[nH]1 C1(F)(C(=O)NC2CCC(C)(CNC(c3ncsc3C3CC3)=O)C2)CC2(CCC2)C1 c1(C(N(CCC#N)CCOC)=O)cccc2c1ccn2CC(C)C c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)CC2F)cc(F)c(Cl)cc1F C1(CC)CN(C)C(=O)CN1C(=O)CC(C(F)F)NC(=O)CCC1CCOC1 C(=O)(C1=CCCCC1C)N(CCN(C(=O)Cc1ccccc1F)CC)CC C12(NC(C3(NC(C(CC)NC(N)=O)=O)CSC3)=O)CC1COC21CCC1 c1(C(=O)OC)cc(C)nc(NC(C2CN(C(=O)C(O)CCSC)CCO2)C)n1 c1(OC)cc(C)nc(N2CCN(C3CCCN(C(=O)C(C)CO)C3)C(=O)C2)n1 C1(C(=O)Nc2cccc(NC(C=CCOCCOC)=O)c2)OC(C)(C)OC1(C)C C(=O)(C(CC(N)=O)NC(=O)C(C#N)C(C)C)NC(c1c(C)ncs1)C CC1(C)OCCN(Cc2ccc(C#N)s2)C1c1ccccc1 N1(C(c2n[nH]c(CC)c2Br)=O)CC2CC(NC(=O)CC=CC(C)(C)C)C1C2 N1(C(c2cnn(CC(=O)OC)c2)C(=O)NCCCCCC)CC2(C1)OC(=O)NC2C N1(C(c2ncnc3c2CCC3)=O)CCCC2(CCCN2C(c2nncs2)=O)C1 C=CC(C)(O)C(=O)NC1CCCC(C(=O)NCCCN(C)C(C)=O)C1 C(=O)(C(CC)CC(C)C)N1CCC(N(C(CSCC=C)=O)CCO)CC1 C1(C(C)NC(c2ccsc2)C)CC12CCC2 c1(C(N2C(CCC(=O)NCC3CCN(C)C3=O)CCCC2)=O)c(C#N)cnn1C C1(CN(C(C2CN(C(C)C)C2)=O)CC)CCN(C(c2cccc(Cl)n2)=O)CC1 C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)N1CC2CN(C(C(CC)OC)=O)CC2C1 c1(C(=O)NCC(CNC(=O)CC2CCNC(=O)C2)OC)cc2sccc2[nH]1 C1(C(=O)NC2COCCOC2)CN(C(=O)CN2CC=CC2)CC1C1CC1 C1(NC(CN(C(C)=O)C)=O)CCC2CC1CN2C(=O)CSc1ccccc1 C12(C(=O)NCC(CC(C)C)NC(C3CCS(=O)(=O)N3)=O)CCCN(CC1)C2 C(C)(C1=CCN(C)CC1)NC(CCC(C)(C)NC(C(CCCOC)C)=O)=O C1(C)(CNC(C(C)=CC2CC2)=O)COCCN(C(=O)CC(CN(C)C)C(F)F)C1 Cc1ccn(CC(=O)NC2CCCC(CN(C)C(C3(C)COC3)=O)C2)c(=O)c1 N1(CC)CCOC2(CCOC2C)C1.c12ccc(cc1[N+](=O)[O-])[nH]2 CC1CN(C2CC2)CC1NC(C1(CNC(=O)CC2COCCOC2)CCCC1)=O c1(C(=O)NC2CN(C(C(=O)NCCC)C)C(C)CC2)cccn2ccnc12 C1(n2cc(-c3ccc(C(=O)O)nn3)nn2)CC(S(=O)(=O)c2ccccc2)C1 N#Cc1ccccc1S(=O)(=O)N1CCC(C(=O)Nc2ncc(C3CC3)cn2)C1 N1(C(Cc2ccc(OC)cn2)=O)CCCN(C(C2CC23CCC3)=O)CC1CO CC1CC(NC(c2coc(C(F)F)c2)=O)CN(C(=O)CNC(C2CCCC2)=O)C1 C1(C(=O)NCC2CC(C)N(C(=O)CS(C)(=O)=O)C2)CC2(C1)CC(C#N)C2 N12CCN(CC1)CC2.C1(CC(=O)N(c2snc(CCC)n2)C)CCOCC1OC c1ccc2c(c1)OCO2.c1cc2cc(c1)C1(CCCC1)N2.c1ncc[nH]1 Cc1ncc(NC(C2CCN(C(c3cnc(Br)o3)=O)CC2O)=O)c(C)n1 c1(CC(=O)NC(C(C)NC(=O)Cn2ccnn2)C)ccccc1-n1cccc1 N1(C(CC(CCC)(C)O)=O)CC2(C1)CN(C(C1CCCOC1)=O)CC(C)(C)O2 C1(C(N(CC(=O)N(C)C)CCC)=O)CC(C)CN(C(c2nnn(C)c2N)=O)C1 N1(C(C=CC)=O)CCC(C(=O)NCc2ccn(-c3ccccc3)n2)C1(C)C Cc1nsc(NC(C2CCN(C(C3(C)CCNC3=O)=O)C2)C)c1C#N C1(CCCC)CN(C(C2C(C)C2(F)F)=O)CCN1C(c1csc(COC)c1)=O c1(C(N2CCC(CO)C(O)C2)=O)ccc2nc(-c3cnc(F)c(F)c3)sc2c1 N1(C(c2n(C)nnc2)=O)CC2CCCC2(NC(C2CCN(CC(F)F)CC2)=O)C1 C1(CNC(c2nc(CC)sc2)=O)N(C(=O)C(C)C#N)CCC1(C)C c1(C(N2C(CNC(CC3CCCC(OC)C3)=O)CC2)=O)nc(C)ncc1Br Cc1cc(C(=O)NCC2(O)CN(C(c3cc(F)n[nH]3)=O)C2)c(C)cc1Br C(CC(=O)NOC(COC)COC)N(CC=C)C(C1CCCC1COC)=O Cc1cc(OCC(=O)NCC#CCNC(C2CC2C2CC2)=O)cc(C)c1 c1(C(=O)NCCCN(C(=O)C(F)=C(C)C)CC)ccc2oc(=O)oc2c1 CC1(C)C(C(N2CC(OCCC(=O)NCC(O)CF)C2)=O)C1(C)C N1(C(C(C)OCC2CC2)=O)CCCN(C(c2cocc2C(N)=O)=O)CC1CO c1(C(N2CC(F)(c3cn(C4CCCC4O)nn3)C2)=O)cc2ccccc2[nH]1 n1(CC)cnnc1CCNC(=O)C(C)N(C(=O)C(C)n1cccn1)C1CC1 N1(C(COCCC=C)=O)CCCC2CN(C(c3csc(C(F)F)n3)=O)CCC12 N1(C(c2c(C)nns2)=O)CC(NC(=O)CNc2ccccc2Cl)C(C)(C)C1 C(=O)(C1COc2ccc(Br)cc21)N(C(C)CNC(c1ccncc1O)=O)C CC1(C)C(CC(=O)N(CCNC(=O)CC2CCCC(O)C2)C2CC2)CC1O Cc1cc(C(=O)N(CC(C)CNC(c2cnn(C(C)C)c2C)=O)C)c(O)nn1 C(=O)(C#CC1CCCC1)N1C(C)C2CC1C2NC(=O)CCn1cccn1 Cc1cc(C(=O)NCCCC2CCCN2C(=O)C(C)n2cncn2)nnc1O Cc1cc(F)c(C(N2CC3CC2CN(C(c2nccs2)=O)C3)=O)cc1Br C(=O)(CCCCCC#N)NC1C(SC)CN(C(c2cnc(C(C)C)[nH]2)=O)C1 Cc1ccnc(CN(c2scc(CC(=O)NCCCCNC=O)n2)C)c1 C=CCCC(C(=O)NCC1CC[Si](C)(C)C1)NC(c1cc(CC)n(C)n1)=O CC(CCCNC(=O)CC(=O)N(C)C)NC(=O)Cc1sccc1Cl CS(=O)(=O)c1ccc(C(N2CC(NC(C3CC34CCOC4)=O)C2)=O)s1 C(CCC(C)(C)C(=O)NCC(=C)CC)NC(COCC(=C)C)=O C(CC(=O)N1CCCC(CC2CC2)C1)(C(C)(C)C)NC(c1c(CC)csc1)=O CCC(F)(F)C(C)(C)C(=O)N1CCC(CNC(c2ncc(Cl)cc2Cl)=O)C(C)C1 CC1CC(N(C(=O)CC2(C)CCN(C(c3cc[nH]n3)=O)C2)C)CCO1 c1(OC)ccc(Cl)c(NC(=O)C(CC#N)c2ccccc2)c1 N1(C(C2(SCC)CC2)=O)CCCCC2(CCN(C(=O)CC3CNC(=O)C3)C2)C1 c1(C(=O)NCCCN(C(=O)C(C)(COC)OC)CC)cc(S(N)(=O)=O)c[nH]1 c1(C(N2C(CNC(C3N(CC)CCOC3)=O)CC2)=O)cnc2c(c1)NC(=O)CO2 C1(C(N2CC3C(NC(C4CCC5CC4CO5)=O)(C3)C2)=O)CC2CCCC(C1)C2 Cc1c(C(N2CC=CC(NC(C3CC34CCC4)=O)C2)=O)ccc2c1CCC2 C1(NC(C(CCOC)C)=O)CCN(CCOC2CCC2)CC1O C1(C)(NC(C2CCN(C(CC=CCC)=O)C2C(C)C)=O)CCC(C)(C)CC1 c1(C(=O)NC2CCCC2C(=O)NCC2CCCC2)cc2[nH]ccc2cc1Cl c1(C2(C(=O)Nc3[nH]nnc3-c3ccccc3)CCC2)ccccc1Cl c1(C(N)=O)cccc(C(=O)NC2CC(O)C2)c1.C12(CC1)C(=O)NC2C1CCC1 Cc1nn(C)c(C)c1OCC(=O)NC1CC(F)(CNC(=O)CCCN(C)C)C1 C1(CC=C)(C(=O)NCC(c2ccccn2)O)CCCN1C(=O)CC1CSC1 C1(COC)(NC(=O)C(F)C(F)(F)F)CCN(C(C2(C3CCCO3)CCC2)=O)CC1 C1(N(C(c2cnc(C(C)C)nc2)C(=O)NCC2CC2)C)CCC2(CC1)CC2 C(=O)(CCCCCCCC)NC1(CO)CCN(C(c2c(CC=C)nn(C)c2)=O)C1 c1(C2CCN(CCCCC(=O)N(CC(=O)O)C)C2)ccc(Cl)c(-c2nn[nH]n2)c1 N1(C(c2c(NC)nccc2)=O)CCC(C2CCN(C(=O)C(C)(C)CO)C2)CC1 C(=O)(CCCCCN(C)C)N1CCC(N(C(=O)C(C)(C)N(C)C)CC(=O)NC)C1 N1(C(CNC(C)=O)=O)CCC(NC(=O)Cc2cc(C)ccc2F)C12CCC2 C(=O)(C1=CCOC1)NCCN(CC(C)O)C(=O)COc1cccc(Br)c1 C(=O)(C(C)(C)C(=O)N(C)C)NC1CC(CCC(=O)N(CCCCC(C)C)C)C1 N1(C(CNC(CCCCC)=O)=O)CC2CCN(C(C3CSCC(=O)N3)=O)CC2C1 CCCCCC(O)C(=O)NCC1(OCC)CCCS(=O)(=O)C1 C1(C(=O)NC2C(CNC(C=C(COC)C)=O)C2)COc2cc(F)ccc2O1 C1(NC(=O)CC2(O)CC2)CCC2(CC1)CN(C(c1cc(C(F)(F)F)n[nH]1)=O)C2 C1(CC(=O)NCC(C(C)C)NC(C2(CO)CCOCC2)=O)CC(C)(C)CO1 N1(C(CC2C(=O)NC(=N)S2)=O)CCC(C2(NC(C3CCC(=O)NC3)=O)CC2)CC1 Cc1cc2cccc(C(=O)NCC3C4CN(C(C)C)CC34)c2[nH]1.c12cnncc1S2 C(=O)(CC(C)CC(C)C)N1C(C(=O)NCC(C(=O)NC)O)CC1C C1(CC#C)(C(=O)NC2CC(NC(c3ccc(NC)cn3)=O)C2)CCCCC1 N1(CC)CCN(C(=O)CC2(C)CCN(C(=O)Cc3cncs3)C2)CC1C C1(OC)CCC(C(=O)NC(CCCNC(C2(Br)CC2)=O)c2ccccc2)CC1 N1(C(c2c(C)ncc(N)c2)=O)CC(NC(=O)C(F)n2ccnc2)CC2(CCC2)C1 c1(NCCN2CCN(C(c3c(C)scc3)=O)CC2)cc(C#N)ccc1O C1(NC(C(C)(C)OCC)=O)CC(NC(=O)Cc2cc(C(=O)OC)cs2)C12CCC2 c1(C(=O)NCCC2(NC(C34CSCC3C4)=O)CCCC2)cccc([N+](=O)[O-])c1 Cc1cc(F)ccc1CC(N1CCC(NC(c2cocn2)=O)C(F)C1)=O c1(C(=O)NCC2N(C(c3c(N)nccc3)=O)CCC2)ccc(Cl)c(Cl)c1 Cc1nc2ccccc2nc1C(=O)NC1CN(C(=O)C2=CCOC2)CCC1C c1(C(C)(C)C)nsc(N)c1C(=O)NC(CNC(=O)CC1CC1(Cl)Cl)CO c1(C(=O)NC(c2cn(CC3CCC3NC3CC3)nn2)=O)cc(C2CC2)oc1C1CC1 c1(OCC)cccc(CCNC(=O)C=CCOc2cccc(Cl)c2)n1 N1(C(C=C(CC)C)=O)CCN(C(C2CCN(C(C)=O)C2)=O)C(CC(F)F)C1 C1(CNC(C2(C#C)CCC2)=O)CN(C(=O)CC2CC(C3CC3)C2)CCO1 N1(C(C(C)(C)OC(C)=O)=O)CC(CNC(=O)CC2CC3(CC3)C2)C(F)(F)C1 C12(C(=O)OC)CCC(C(=O)NCC(C)NC(c3sccc3C#N)=O)(COC1)C2 C(=O)(C(C)CC(F)F)NC1CC(NC(CSc2ccc(OCC)cc2)=O)C1 Cc1ccc(O)c(C(=O)NCC23CC2CN(C(C2CCCN(C)C2)=O)C3)n1 C1(C2(O)CCN(c3ncnc4c3COC4)CC2)(NC(c2c[nH]c(=O)cn2)=O)CC1 CC1C(=O)CCC(C(=O)OCCc2ccccc2F)C1(C)C N1(C(c2cc(OC)no2)=O)CC2(CC(NC(=O)CC3CCCCC3O)C2)C1 c1(C2(C(=O)NC(C)CNC(c3coc(Cl)n3)=O)CC2CO)cccc(Cl)c1 N1(C(c2ccc(SCCC)cc2)=O)CCN(C(C2CCC2C)=O)C(CO)C1 c1(OC)ccc(C(=O)NC2(C)CN(C(=O)Cc3cnccc3C)C2)cc1C(C)C c1(N2CCCC(CC=C)(NC(=O)C(C)CCC)C2)nc(C)cc(C)c1C#N c1(C(N2CCC(NC(C3(C)C=CCCC3)=O)C(F)C2)=O)nc(O)nc(O)c1N C(c1cn(C)nn1)=CC(=O)NCC(C)NC(CNC(CC)=O)=O c1(C(N2CCN(C(CC(C(C)C)O)=O)C(CO)C2)=O)noc2c1CCCC2 c1(NC(C(CNC(C2CC=CCC2C)=O)OC)=O)cc(F)ccc1C C1(NCc2nc(N(c3cccc(C4CC4)c3)C(C)=O)sc2)CN(C)CCO1 c1(C(N2CC(C)C(CNC(C3(C)CCNC(=O)C3)=O)C2)=O)ncsc1S(N)(=O)=O S(=O)(=O)(c1ccc(N2CCC3(CCCC3)C2)cc1Br)NCC1(OC)CCSC1 C(=O)(C1=NN(C)C(=O)CC1)N(C1CCN(C2CCCC2O)CC1)C N1(C(C=C(C)C(C)(C)C)=O)CCC2(CCC2NC(c2cc(Cl)ns2)=O)CC1 Cc1ncc2cc(C(=O)N(C3CCC(NC(C4CC4[N+](=O)[O-])=O)CC3)C)ccn12 c1(CC(=O)NC2CC2CNC(C2(O)CCOC2)=O)ccc2ncccc2c1 CON1CCC(C(=O)NC(C)C(C)C(=O)NCCC(=O)NC(C)C)CC1 C1(CNC(C2N(C)CCCCC2)=O)CN(C(C2CC2C(F)F)=O)C2(CCC2)C1 C1(CCN(C(C(CN(CC)CC)F)=O)C)CCCCN1C(c1cccc(Cl)c1)=O N1(C(C=CCOCCOC)=O)CCN(C(c2cnc(O)s2)=O)CC1c1nccn1C c1(C(=O)NC2CCCC(CNC(C3N(CC)CC3)=O)C2)c(OC)ccc(Cl)c1Cl N1(C(c2c(C)cno2)=O)CCC(NC(c2scnc2Cl)=O)C1c1ccccc1 N1(C(C(C)CN(C)C)=O)CCC(C)(C)C1C(=O)NC1CN(c2ncco2)C1 N1(C(C2C(C)C2C)=O)CCCC2(CCCCC2NC(=O)CC2CCCCCC2)C1 Cc1ccsc1C=CC(=O)NC(C1CCCN1C(C1CCCN1C1CC1)=O)(C)C C(C(=O)NC1CN(C(=O)C=C(C)Cl)CC1SC)(C(C)C)NC(C)=O C1(C)(C(=O)NC(C)CN2CCCC2)CCN(C(=O)Cc2cnoc2)CC1 O=C(C1(c2cccs2)OCCN1C(c1ccccc1)=O)OC.C12(CC=O)CC(C1)C2 Cc1cnn(CC(=O)NC(C)(C(=O)N(C(CF)CF)C)C2CCC2)c1 c1(C(=O)NC2CC(CCNC(=O)CC3CCCCO3)C2)cccc2[nH]ncc12 c1(C(=O)NCCCN(C(C(F)=CCC)=O)CC)ccc(-n2cncn2)cn1 C1(N(C(C(CC)=CC)=O)C)CCC2CN(C(=O)Cc3nccn3C)CC12 C1(S(=O)(=O)Nc2ccccc2N(C)C)(c2cn(C(C)COC(F)F)nn2)CC1 C(=O)(C(C)C(=O)NC(C1CC1C(=O)NCC#CCCO)C)OC C1(C(N2CCC(C3CCCCN3C(c3ccsc3)=O)C2)=O)CCCC(F)(F)C1 N1(C(CCSCC(N)=O)=O)CCC(NC(=O)CC2CC(F)C2)C(O)C1 c1(OC)cccc2cc(NC(C3CN(C)CC3c3ccccc3)=O)cnc12 c1(C(=O)NC2CCC(NC(CCCC=C)=O)CC2)cn(C)c(=O)n(C)c1=O c1(C(=O)NCC2(N(C)C(c3ccc(C4(C)CC4)cc3)=O)CC2)cc(O)cc(Cl)c1 N1(C(C(N2CCCC(C)C2)=O)=O)CC(NC(=O)C=Cc2ncc[nH]2)CCC(O)C1 C(c1ccco1)=C(C)C(=O)NCC1CC(NC(=O)CNC(C2(C)CCCO2)=O)C1 C(=O)(CC(C)(C)C(F)F)NC(C)CCNC(=O)CC1(C)CC1(Cl)Cl C1(n2cc(C3(C)CC3)nn2)CCCN(CC=CCC(N2CCCCC2)=O)CC1 C(=O)(CCCCCCNC(=O)CCC1CC(OC)C1)NCC1(C#C)CCCC1 C(CCCCC(=O)N1CCC(NS(C)(=O)=O)C1)n1cc(-c2nc(C)sc2)nn1 C(=O)(C1=COCCC1)NCc1cccc(CNC(C2(C)CC2Br)=O)c1 C(=O)(C(C)P(C)(C)=O)NCC(C(C)C)NC(c1cnc(-c2ccccn2)s1)=O c1(C(=O)NC(CC=C)CNC(C2(C(C)(C)C)CCC2)=O)cnc2cccnc2c1 C=CCC(C)(C)C(=O)N1CCN(CC(C)(C)NC(C2(OC)CCCC2)=O)CC1 N1(C(=O)CC2CCCCCC2)CC2CCC(CNC(=O)C(F)(F)CO)(C2)C1 c1(NC)cccc(C(=O)NCCCN(CCCNC(=O)C=CSc2nc[nH]n2)C)n1 N1(C(COCCOCC)=O)CCN(C(c2ccnn2C(C)C)=O)CC1CCOC CC(C)C(CCN(C)C(c1ccno1)=O)NC(c1cc(-n2cccc2)ccn1)=O C1(NC(C2(F)CCN(C(C(CC)(C)OC)=O)C2)=O)CCC(C2CC2)CC1 Cc1ccc(C2CC2)c(C(=O)NC2CC3(C2)CN(C(=O)C(F)=CCCF)C3)c1 Cc1nn(C)c(C)c1CCC(N1CC2CC(C1)C2NC(=O)CC(C)(C)C)=O O(NC(=O)C(CC(=C)C)NC(C1CCC(=O)O1)=O)CCCC#C CC1CCN(C(=O)CCn2cc(Cl)cn2)CCN1C(C1CCN(C(N)=O)CC1)=O c1(CC)cnc(N2CCOC(CCC(=O)OC)C2)nc1 C(=O)(C(F)(F)CO)NCC(c1ccc(F)cc1)NC(c1cc(SC)oc1)=O C1(c2ccc(F)cc2)(C(=O)NC(CC)CNC(c2[nH]ccc2C)=O)CCOCC1 C12(CNC(=O)C(C3(O)CN(C(=O)CC4CC5(CCC5)C4)C3)F)COC(CF)(C1)C2 C(=O)(C1=C(F)CN(C(c2cnsn2)=O)CC1)N(CC=C)CCC c1(OC)ccc([N+](=O)[O-])c(N2CCC(CCOC(c3ccccc3)=O)C2)n1 c1(C(N2C3CN(C(c4cccc(OC(F)F)c4)=O)CC23)=O)cc(F)cc(Cl)c1C c1(OC)ccc(F)cc1C(=O)NCC1C(C)CCN1C(c1ccc(Br)o1)=O C1(C(=O)NC(c2ccccc2O)C)CN(C(c2cnsn2)=O)C(C)(C)C1 CC1(C)CCN(C(=O)COCCc2ccccc2)CC1CNC(=O)C1=CCSC1 c1(C(N2CC3CCN(C(C(CCC)C#N)=O)C3C2)=O)cc2cc(C)ccc2o1 C(=O)(C#CC1(C)CCCO1)NCC1(NC(c2cc(C3(C)CC3)on2)=O)CC1 c1(NC(COC)=O)cccc(C2(C)CC2)c1.C1(=O)C(=O)NC1.C12(CC1)C(C)C2 C(=O)(C1=CC2CCC1C2)N1CCC(CN(C(CCc2ccc(C)cc2C)=O)C)C1 n1(CC(=C)C)c(N2CC3C(COC)C3C2)nnc1COCC c1(C(C(=O)NC(CC(=O)NC)C)NC(C2CSCC(=O)N2)=O)c(C)cccc1Br c1(C(N(CC(C)NC(CCCCOCC)=O)C)=O)cc(OC)c2c(c1)OCO2 CC(C)C(F)(CNC(C1(C)C=CCC1)=O)C(=O)NCC(=O)N(C)C c1(CNC(COC(C)=O)=O)nnn(C)c1C(=O)NCC1COC(CO)C1 c1(C(=O)NC(C)CN(C(=O)CCn2ccc(=N)[nH]2)C)cc(C2CC2)ccc1F N1(C(CS(=O)(=O)NC)=O)CCC2(C1)CN(C(c1c(C)nsc1Cl)=O)C2 C1(CC)CCOC1C(=O)NC1CCC1C(=O)NCCCNC(=O)OC c1(C(=O)NCCCCNC(C2CC2C(F)F)=O)cc2n(n1)CCNC2=O CC(CC(N)=O)C(=O)NC(C)CCN(C(=O)C(F)(F)CCn1cccn1)C Cc1ccc(C(=O)NC(CNC(=O)CC(C)C2CC2)CC(C)C)c2c1CCC2 Cc1cc(N2CC3C(C(=O)N(C)CCOCCCC(C)C)C3C2)nc(C)c1 N1(C(c2c(OC)n[nH]c2)=O)CC(NC(=O)C(C)C(F)F)C(O)C1 C1(CC(=O)NCCCOCCNC(C2CCCOCC2)=O)CCC12CCC2 C(=O)(C(C)(O)CCN(C)C)OC(C)C(=O)NCC(C)(C)S(C)(=O)=O c1(C(CNC(C(CC)(F)F)=O)NC(=O)C2=CCSC2)ccc(Cl)cc1Cl S(=O)(=O)(c1cc(C2OCCO2)ccc1Cl)N(C)Cc1c(C#N)nnc2ccccc12 N1(C(c2ccnc3ncccc23)=O)CC(C2CCCN(C(C3CC(F)C3)=O)C2)C1 C1(C)(C(=O)NCC2N(C(CCc3cc(OC)no3)=O)CC2)CCCCC1(F)F CCCC(C)(O)CC(=O)N1CCC(NC(=O)CC2CC3CC3C2)C(CO)CC1 CC1CC(C(=O)NCC2CN(C(=O)C(C3CCCO3)C3CC3)CCO2)CCN1C c1(C(N2C3CN(C(CCC4C(C)C4)=O)C(C3)C2)=O)cc2n(n1)CCNC2=O N1(C(c2c(C)nns2)C(=O)NCCC2(C)CC2)CC2(CCCC2)OCC1C N1(C(C(C)C2CCC2)=O)CC=C(CNC(=O)Cn2ccc([N+](=O)[O-])n2)CC1 C12(C(N(C(CC)C)CCO)=O)CCCC1CN(C(c1[nH]nnc1C)=O)C2 C1(C(=O)NC(C)(CNC(C2(n3cccn3)CC2)=O)C2CCC2)CCC(F)(F)C1 N1(C(COCC(=O)OC)=O)CC2(CCCC2NC(=O)C(C)Cc2c(C)noc2C)C1 C1(NC(c2c(C)n(C3CC3)nc2)=O)CCN(C(c2cc(Cl)no2)=O)CC1CO N1(C(CCC(=C)C)=O)CCCC(N(C)C(C2CC(Cl)(Cl)C2)=O)CC1 C1(CC(=O)NCC(C#C)OC)N(C(=O)CC2CCCC23CC3)CCC1(C)C N1(C(C2CCN(CCC)CC2)=O)CC2CCOC2(CNC(C2(CC)CCC2)=O)C1 CCCCCCCCC(=O)NC1CCC2(CCN(C(C3C=C(C)CS3)=O)C2)C1 N1(C(CC2C(CC)C2)=O)CCCC(O)(CNC(c2nccc(Cl)c2O)=O)C1 CC(C)CCC(=O)NC(C)(C)CCNC(=O)CCC1CC1CC1CC1 N1(C(C(COCC)NC(C2(n3cnnn3)CC2)=O)=O)CC2CCC(O)C2C1 CCCCC(C)(F)C(=O)NC1CC1NC(=O)Cc1cncnc1O C1(CNC(c2cscn2)=O)CCCCN1C(=O)CC1CCC2CC12 c1(C(N2CCCC(F)(CNC(C3CC3C3CCC3)=O)C2)=O)cccc2sccc12 C1(CC=C)NC(=O)CCN(CCc2cn3cccc(C)c3n2)C1=O N1(C(C2(SC)CCC2)=O)C2CCCC1CN(C(=O)C(C)SC(F)(F)F)CC2 N12C3CCC1C(C3)C2=O.CCS(=O)(=O)NC(=O)C(=O)NC(C)C c1(NC(N2CC(C(=O)Nc3cccc(C)c3)C(C)C2)=O)ccc(C)c(C)c1 Cc1cc(C(=O)NC2CC(NC(=O)C(C(C)C)NCc3ccco3)C2)nc(O)n1 c1(N(C(=O)C(c2ccccc2)NC(=O)C(N)CCC2CC2)C)cc(F)ccc1N c1(C(=O)NC(CN(C(=O)C(C)N(C)C)CC)C)sccc1C1CC1 c1(C(=O)NCC(C(C)(C)C)NC(CC=C=C)=O)cc(Cl)ccc1OC(F)F CN1CC(O)CC1(C)C(=O)NOCC(=O)NCC1(F)CC=CCC1 c1(CC)ccc(O)c(NC(=O)COCCNC(=O)C(C)(F)F)c1 C1(CNC(CCCCCC)=O)C(C2CC2)CCN1C(c1cc(Cl)no1)=O C1(C#N)(C(N2CCC(CC=C)(NC(c3sc(F)cc3C)=O)C2)=O)CC2CC2C1 C12(CCNC(C(C)(C)c3cscn3)=O)CCC1CN(C(c1cccnc1O)=O)C2 CC1(C)CC(NC(C2CC(OC3CC3)C2)=O)CN1C(=O)CSc1n[nH]c(O)n1 O=C(CS(=O)CCC(F)(F)F)NNC(=O)c1cccc(Br)c1 C(CCC(C(=O)N1CCC(OCCO)CC1)NC(c1cncn(C)c1=O)=O)OC c1(NC(c2cc(CSC)no2)=O)cccc2ccccc12.C1(C(=O)N)(CO)CCCO1 C1(N(C(C2CN(CC(C)C)C2)=O)C)CCCCN(C(=O)CCC2CCOC2)C1 c1(C2(C(=O)NC(CNC(COCC#C)=O)C)CCC2)ccc(Cl)c(Cl)c1 C1(NC(C2CC(C)(NC(C(C)CC3CCCC3)=O)C2)=O)CC12CCCCC2 c1(NCCCCOC(C)C)ccc(S(=O)(=O)N2CCOC(CCN(C)C)C2)cc1Cl C1(C(=O)NCCC2(CNC(C(CC)N(C)C)=O)CC2)CC(C)(C)OC1(C)C CC1CC(C(N2CCSCC2C2CC2)=O)CCN1 N1(C(C2CCC(C)(C)O2)=O)CCCC(O)(CNC(C2CC(F)C2)=O)C1 Cc1cc(N2CCCC(c3cnc[nH]3)C2)cnc1F Cc1csc(C=CC(N2CC(NC(=O)C(O)C3CC3)C(C)C2)=O)n1 N1(C(C2CC(SC)C2)=O)CCN(C(=O)Cc2cc(C(F)F)on2)CC1 c1(C(N(CC(C)N(C(=O)C2=CSCCO2)C)C)=O)cccc2c1ccn2C c1(C2C(C(=O)NC(CNC(CCOCCC)=O)CO)C2)ccc(F)cc1 N1(C(COCC(=O)OC)=O)CC2=C(C1)CN(C(c1c[nH]c(=O)c3ccnn13)=O)C2 c1(NCC2C(C)(C)OC(=O)C2)ccc2c(c1)CCC(=O)N2 CC1CCC(NC(c2coc(C(F)F)n2)=O)CN1Cc1ncc(Cl)n1C C(=O)(CS(=O)CCC(F)(F)F)N(C1(c2nn[nH]n2)CCSC1)C C1(NC(C(COC(C)C)NC(C2CCC(CC)CC2)=O)=O)CCC(C)(O)CC1 CCCCC(C)C(=O)NCC1(CNC(Cn2ccnc2)C(C)C)CCCCC1 c1(OCC)cc(C(=O)OCC)cc(CCOC(=O)C(C)CC2CCCC2)c1 C(=O)(CC1=NN(C)C(=O)C1)NC1C2C(NC(CC(C)C(F)F)=O)CC(CC2)C1 S(=O)(=O)(c1cccc(CO)c1)NC(C1CN(C(C2N(C)CCC2)=O)CC(F)C1)=O c1(SC)cccc(C(=O)NCC(C)CNC(c2sc(-c3ncc[nH]3)nc2C)=O)c1 C1(C)(NC(c2n(C)c(Cl)nc2)=O)CCCCC1C(=O)NCCCc1cncnc1 N1(C(Cc2ccc(OC)cn2)=O)CCC2C(CCCN2C(=O)C=Cc2cc[nH]c2)C1 C1(C(N2CCC(OCCNC(c3n(C)ncc3Cl)=O)CC2)=O)CCOC(C)(C)C1 CC(C)(CC(F)F)C(=O)NCC1CC(NC(=O)CCC2CCCCCC2)C1 C1(CC)C(NC(C2(C)CS(=O)(=O)C2)=O)CCN1C(=O)CNC(=O)NC c1(OC)cc(CNC2CCNCC2c2ccccc2)cc(OC)c1Br c1(C(N2CCN(C(C3(CO)CC3)=O)CC2C2CC2)=O)cccc(Cl)c1Br c1(C(=O)NC2(C(=O)NC3CC(CC)C3)CSC2)cc(CO)[nH]n1 CC1(C)C(CNC(c2ncc(C(F)(F)F)s2)=O)CCN1C(C1CC12CC2)=O C1(CNC(CC2(C=C)CC2)=O)CN(C(C2CC(=O)N(CC)C2)=O)CC12CC2 N1(C(C2CC(=C)C2)=O)CCN(C(C2CCC3(CC3)C2)=O)CC1C C1(C(=O)NCC(C(C)C)NC(c2cccc(N)c2)=O)CC2C=CC1CCC2 N1(C(CC2ON=C(C)C2)=O)CC2(C=C(C(=O)NCC(F)F)CO2)C1 C1(NC(C(C)NC(N)=O)=O)CN(C(C2C(C)(C)C2(F)F)=O)C2(CCCCC2)C1 c1(OC)cc(C)c2cc(C(=O)NC3(C)CN(C(=O)CCOC(C)CC(C)C)C3)[nH]c2c1 C1(C)(CNC(=O)NC(c2ncc[nH]2)CC)CCN(C)C1 c1(SC2CC(CNC(c3cccc(OC)c3)C(=O)OC)C2(C)C)ccc(Br)cc1 C1(OC)CCN(C(c2csc(Br)c2)C(=O)NCCCF)CC1 C(=O)(n1nccc1NC(c1ncsc1Br)c1nnnn1Cc1cccs1)N(C)C C1(C(=O)NC(CN(C(c2coc(Br)n2)=O)CC)C)COCCO1 C1(F)(C(=O)OC)CCCN(C(=O)C(C(C)C)OC(c2cc(C)cc(C)c2)=O)C1 N1(C(Cc2nc(C)[nH]n2)=O)CC(CCNC(=O)C(C)(C)c2cnco2)C(C)C1 CN1C2CCC1CC(C(=O)NCC1CN(C(c3cc(C4CC4)on3)=O)CCO1)C2 C1(C)(C(N(C)CC2CCN(C(=O)Cc3cc[nH]c(=N)c3)C2)=O)CCC(=O)N(C)C1 N1(C(C(C)(C)OC(C)=O)=O)CC2CCCC(C1)N2C(C12CCCC1CC2)=O CC(Cn1cccn1)C(=O)NCCCN(C(=O)CNS(C)(=O)=O)C N1(C(c2cncc(C)c2)=O)CC2(CCC2)CC1C(=O)NCc1c(C)n[nH]c1C C1(CC#C)(C(N2CCC(CCNC(=O)CN(C)C3CC3)C2)=O)CCCC1 C#CCCCCCC(=O)NC(C)(CNC(c1nccn1C)=O)C(C)C C(=O)(NNc1nc2c3c(sc2n1C)CC(C)CC3)c1c(C)coc1 C1(CN(CC(C)C)C)CC(C)(C)C1c1ccccc1 C(=O)(CCCC(=O)NC(C)C)N1CC2C(NC(Cc3c(C)cnn3C)=O)C2C1 Cc1cccc(C(C)(C)CNC(=O)C(CO)NC(=O)OC(C)(C)C)n1 Cc1cccc(Cl)c1C(=O)NC1COC2(CNC(c3cc[nH]c3)=O)CC1C2 C1(C(=O)NCCCNC(CC=CC=C)=O)CCCN(C(=O)C(=O)N(C)C)C1 Cc1c(C(=O)N(C2CCCC(NC(=O)Cc3cccnc3)C2)C)cncc1Cl c1(CC)nc(-n2cccc2)sc1C(=O)NCC(F)CNC(c1ccc(F)o1)=O C1(c2cc(Cl)cc(OC)c2Cl)C2=C(N(C)C(=O)N1C)C(C)(C)N(C)C2=O CCC(CNC(c1cccc(C)n1)=O)(CC)NC(c1cc(C(C)C)oc1C)=O C(C(=O)N(CCC(N1CCC(n2cncn2)C1)=O)C(C)C)(C(C)(C)C)OC C=C=CCCC(=O)N1CC(C)(NC(C2C(C(F)F)C2(C)C)=O)C1 C1(CC(=O)N(CCN(C(C2(COC)C=CCC2)=O)C)C)CCCS1(=O)=O c1(N(C)CC)ccc(-c2nc(CC(C)(C)CO)nn2CCS(C)(=O)=O)cc1 C1(NC(C2COCCO2)=O)CCCN(C(=O)CCc2cnoc2)C1 N1(C(C(=O)COC(F)(F)F)=O)CCC(CC(C)C)CC1.C1(CCCN)(C(=O)OC)CC1 C1(CNC(Cc2c(C)nsc2)=O)CCC(C)CN1C(c1cscn1)=O Cc1c(C(=O)NC2CC(CNC(c3c(C4CC4)cnn3C)=O)C2)cnn1C c1(CC)occ(C)c1C(N1CCC=CC1C(=O)NCC(O)C(C)(C)O)=O Cc1ccc([N+](=O)[O-])c(NC(C2C3CC2N(Cc2cnc(C4CC4)s2)C3)=O)n1 C1(NC(COCC(=C)C)=O)CCN(C)C12CCCN(C(c1cnc(=N)[nH]c1)=O)C2 c1(C(=O)NCCN(C)C)cccc(CNC2CC(CO)C2)n1 c1(C(=O)NC2CC(NC(C(CC)OC)=O)CC2O)ccc(F)c(Cl)c1 CC1(CNC(C2(CF)CCN(C(C3CNC(=O)O3)=O)C2)=O)NC(=O)NC1=O N1(C(C(C)(C)C2CCCN2C(=O)C=Cc2cnccn2)=O)CCCC(COC)C1 CCCC(=O)N(C(C)CNC(=O)C(C)O)CC Cc1cccc(C)c1OCC(=O)NCC1(F)CCC(NC(=O)Cn2ncnn2)C1 N1(C(c2ccc(C(C)=O)s2)=O)CCCCC1CN(C)C(c1cnc(C(N)=O)s1)=O C1(CC=C)(NC(c2sccc2C)=O)CCN(C(=O)Cc2cccs2)C1 Cc1nc(C(=O)NC(C2(c3ccc(Cl)cc3)CC2)C)ccc1C(F)F C1(NC(CC2(C(=O)OC)CC2)=O)CN(C(=O)CCc2ccccn2)C2CCCCC12 C1(NC(CNC(=O)NC)=O)CC(C(=O)N(C)CC2CCN(C)C2)C1(C)C N1(C(C2CC(=O)NC2)=O)CC(C2CN(C(c3csc(-c4cc[nH]n4)c3)=O)C2)C1 N(C(=NCC#Cc1cnn(C)c1)NC1CCS(=O)(=O)C1)CC(CC)C(C)(F)F C1(C(N(CCNC(Cc2c(C)scc2)=O)Cc2ccccc2)=O)CC(O)C(=O)N1 c1(C(N(CCNC(c2cscc2Cl)=O)CC2CC2)=O)csc(O)n1 N1(C(C(CN(C)C)NC(c2cc(OC)no2)=O)=O)CC2C(=O)NC(=O)C2C1 c1(CCN2C(CC(=O)OC)CCC2)ccc(Cl)nc1 C1(CC(=O)NC2CCCC2F)CCCC(NC(C2CC3(CC3)CO2)=O)C1 c1(OC)ccc(C(C(=O)N(C2CCN(C(=O)CN3CCCC3=O)C2)C)SC)cc1 C(CC(CC)C(=O)NCC(CC(C)C)NC(=O)CN(C)C(C)=O)=CC C=CCCCC(C1CC1)NC(=O)C(Cn1cncn1)NC(=O)C(C)n1cccc1 S(=O)(=O)(c1ccc(C(=O)N=c2cc(F)n(C)[nH]2)cc1)N1CC(CC)N(C)CC1 N1(C(c2c(CC=C)cccc2)=O)CC(C(=O)NC(c2nncs2)C)CC12CCC2 c1(OC)cc(C(=O)N(C2CCC(NC(C3(C)CC3F)=O)CC2)C)c(F)c(Cl)c1 c1(NC(C(=O)NCCOCC2CC2)=O)ncoc1C1CC1 C=CCC(CC=C)C(=O)N1CC(O)(C2CCCN2C(=O)CC2CCC(C)CO2)C1 C(=O)(CC(C)CCC(=O)NCC(O)CNC(c1cnn(C(C)(C)C)c1C)=O)OC C1(F)(N(C)C)CCN(C(C2(C)CN(C(=O)CCc3cncn3C)C2)=O)C1 C(C)(CCC#N)(c1nnnn1CC1CCCO1)N(C)CCNC(C1CC12CCC2)=O C1(NC(CC(=O)OC)=O)CCCCC1NC(=O)CSS(C)(=O)=O CCC(CC)(CC)C(=O)NC1COCC1CNC(=O)CC1CCCNC(=O)C1 C1(C(=O)NCC(CN(C(C2(CCCC)CC2)=O)C)(C)C)CC2CC(O)C(C1)C2 C(CCC(C)(C)C(=O)NC(C)Cc1cn[nH]c1)NC(C1=C(C)CCC1)=O CC1CC(NC(c2cc(Cl)cs2)=O)CN1C(C1CC(Cl)(Cl)C1)=O CC1(C#N)CCCN(C(C2CC(O)(CNC(=O)CCCCC#N)C2)=O)C1 c1(SCC(=O)NC(C)C(CO)NC(=O)C(c2cccnc2)C)ccc(C#N)cc1 C12(NC(CCCNC(=O)OCC)=O)CCCN(C(C3(C#N)CC=CC3)=O)CC1C2 CC1(C)CCCCC(C(N2CC(NC(C3CC(F)C3)=O)C2)=O)C1 C1(N(C)C(N2CCCC2C(O)C(F)(F)F)=O)CCCN(c2ccnn2C)C1=O C1(C(=O)NCC(C2CC(F)(F)C2)=O)CC(F)(c2ccccc2)C1 N1(C(C2(CC)CC2)=O)CCOCC1CC(N1CC(O)(C(F)F)C1)=O c1(CN(c2ncc(CCC)cn2)CC2CNCCO2)c(Cl)cccc1B(O)O N1(C(C=CC(CC)=CC)=O)CCS(=O)(=O)C(CCNC(c2ccc[nH]2)=O)C1 N1(C(c2cc(C(C)C)no2)=O)CC(CNC(=O)CN2CCNC(=O)C2)CCC1C N1(C(C)C)CC2CN(C(C3CCc4nc(C(F)(F)F)cn4C3)=O)CCN2C1=O C12(C(N(CC(=O)NC)C)=O)CC(CO)(CN1C(=O)Cn1cnnn1)C2 c1(-c2c(C)nc(OC(C)C)cc2)cnc2c(C(N3CCC3CO)=O)c[nH]c2c1 CC(F)(F)C(C)(C)CNC(=NCCF)NCC1CC12CCOC2 N1(S(CCC)(=O)=O)CCCC(NC(c2nccn2C)=O)C1 c1(C(=O)NCC(CCC)C(=O)N2CCC(F)C2)ccc(C#N)cc1C c1(CNC(c2n(CCOCC)nnn2)c2csc(C(=O)OC)c2)nc(C)c(C)s1 C1(NC(c2c(OCC)n[nH]c2)=O)CCCC12CCN(C(=O)C(C)(CC)CO)CC2 C(C(=O)NC1CN(C(=O)CCN(C(=O)CO)C2CC2)C1)(C(F)(F)F)OC(C)(C)C n1(CC)nnc2c1CCC(C(=O)Nc1ccc(SC(F)(F)F)nc1)C2 Cc1scnc1C(N1CC(C)(NC(=O)Cn2cc(CN(C)C)nn2)C1)=O c1(C(N2CCC(O)(CNC(c3cc(C)nn3C)=O)C2)=O)c(C)nn2ccccc12 C1(NC(C2CCN(CC)C2)=O)CC2CN(C(c3cc(OC)cc(F)c3)=O)CC2C1 c1(CCC)nsc(N)c1C(=O)NC1(CNC(c2csnc2C)=O)CC1 N1(C(c2ncc(N(C)CC)s2)C(=O)NC2CCCC2)CCCS(=O)(=O)CC1C.CC N1(C(C(CC=CCC)C)=O)CCN(C(c2cnc(C3CCOC3)s2)=O)C(C)C1 C1(=O)C(C(C)C)N1.c1(C(=O)NC2CC(COC)C2)cc(C(F)F)[nH]n1 c1(C(=O)NC2CC(C)N(C(=O)CCC3CCC(O)CC3)C2)cc(Cl)c(N)c(Cl)c1 CC1(CNC(c2scnc2C(F)(F)F)=O)CCCN(C(C2CC23CCCC3)=O)C1 n1(CCNC(Cn2cc(C(=O)OC)nc2)=O)cc(C#N)ccc1=O c1(CC)oc2ccccc2c1C(=O)NCCN(CC(C)O)C(c1cc(C)nn1C)=O c1(NC(C2N(Cc3ccc(C(=O)O)[nH]3)CC3(CC3)C2)=O)nc(Cl)c(Br)cc1O c1(C(=O)NCC2(CNC(c3ccc(=O)n(CCF)n3)=O)CC2)c(O)cccc1Cl C1(NC(C(C)S(C)(=O)=O)=O)CC2(CCC(CNC(=O)CC3CC4CC4C3)CC2)C1 C1(C2CCN(C(=O)Cc3ccc(Cl)c(Cl)c3)CC2)(NC(C2C(C)C2)=O)CC1 N1(C(C(CCSC)NC(CNC(CCC)=O)=O)=O)CC(O)C(C2CC2)C1 c1(OC)c(Cl)cc(CN(C)C(=O)NC(c2cccc(C(F)(F)F)c2)C)cc1Cl c1(C(=O)NCCN(CCCCCC)C(c2cscn2)=O)cc(O)c2sccc2c1 C1(CC)CCCCC1C(N1CC(NC(c2ccoc2CC)=O)CC1C)=O C1(F)(NC(=O)NCCN2CCC(CC3CC3)C2)CCCCC1 c1(C(=O)NCC2(CNC(C3CCC(C)S3)=O)CCC2)ccc(C(F)F)c(F)c1 c1(NC(=O)NCCNC2(CCC=C)CC2)cc([N+](=O)[O-])c(C)s1 C1(C(=O)NCC2(F)CCCN(C(C3(F)CC=CC3)=O)C2)CC2(C1)CC1(CCC1)C2 c1(C(=O)NC2CCN(Cc3cn(CC(=C)CC)nn3)C2)ccc(Br)cc1Cl c1(C(N(CCNC(c2noc(CC)c2C)=O)CC)=O)cc(C)c(O)nn1 CC1(C)CN(C(C2CCCSC2)=O)CC2(CN(C(C3CCC34CCC4)=O)C2)O1 c1(C(C)(C)C)ccc(C(=O)NC2CC(C(=O)NC3CCCC3C#N)C2)nc1 CCCCC(CC)CC(=O)NCC1(C)CN(c2ncnc3[nH]cnc23)CCO1 C(=O)(C(CC)NC(C)=O)NC1CCC(NC(CC)=O)C1 C(CC(=O)NCCOC1CCN(C(C2CC23CCOC3)=O)C1)(C(F)(F)F)OC N1(C(C(C)CC2CC2)=O)CC2(C1)SCCC2NC(=O)CCCc1ccncc1 S(=O)(=O)(c1cccc(=NC(CC2CCCO2)CO)[nH]1)CCCN1C(=O)CCC1 C1(N(C)C(C23CCC(CC2)C3)=O)CC2CC1N(C(c1csc(NC=O)n1)=O)C2 C1(C(N(C2CCCCC2NC(=O)COC2CCCCC2)C)=O)COCCN1C=O CS(=O)(=O)C1(C(N2CC=C(CNC(=O)CC3CCCCC3)CC2)=O)CCCCC1 c1(C(=O)NC2CCN(C(c3c[nH]ccc3=O)=O)CC2CO)noc2c1CCCC2 c1(C(=O)NCC(c2ccccc2)NC(C2(O)C(C)(C)C2)=O)cn2ccnc2s1 c1(CNC2C(C(N3CCCC(O)C3)=O)C2)c(F)cc(I)cc1F CC1CN(C(c2sccc2OC(F)F)=O)CC(CCNC(C2(O)CCC2)=O)O1 c1(C(=O)NC2CN(C(Cc3c(C)ccc(C)c3)=O)CC2C)cc([N+](=O)[O-])c(C)s1 C1(CC)(CC)CC(NC(c2cnc(C)n2C)=O)CN1C(c1cc2occc2[nH]1)=O CC1CCN(C(=O)CC2CC3(C2)CN(C(C2CC(=O)CS2)=O)C3)C(C)C1 C#Cc1ccc(C(N2CC3(CCN(C(c4scnc4C)=O)C3)C2)=O)cc1Cl c1(OC)cccc(C(F)(F)F)c1C(=O)NC1CN(C(=O)C2=CCCS2)CCC1CO c1(C(N(C2CCN(C(c3snnc3CCC)=O)CC2)CC#C)=O)[nH]c(C)nc1C c1(C(=O)NCCC23C(CN(C(CCCC)=O)C2)CC3)cnc(O)c2ccsc12 c1(NC(C(CCC)C)=O)ccc(NC(=O)C(c2ccccc2)N(C)CC)c(C)c1 O=C(C1=CCCOC1)NC1CCOCC1C(=O)NC1(C2CC2)CC1 c1(C(=O)NC(C(CC)CC)C(=O)O)ccc2c(=O)n(C)c(S)nc2c1 N1(C(c2cc(CCC)on2)=O)CC(CNC(C2CN(C(C)C)C2)=O)CC(C)(C)C1 C1(C(=O)NCCC2CC(NC(c3c(C(C)C)nccc3)=O)C2)CC12CCCOC2 C1(NC(CSCC#C)=O)CCC(CNC(c2csc(C(F)F)c2)=O)C1 c1(C(N(C)C)=O)cc(NC(C2CC3CC3N2c2ncccn2)=O)cc(F)c1 C1(C(=O)OC(c2cccc(Br)n2)C(=O)OC)COC(C)CO1 C(C(C(=O)NC1CC(CCC(=O)O)C1)n1cc(CC(O)C(C)C)nn1)OCC c1(OC)ccc(NC(c2n[nH]c(C)c2C(F)(F)F)=O)c2cccnc12 S(=O)(=O)(c1c(Oc2c[nH]c3cccc(OC)c32)ccc(Cl)c1F)OC(F)(F)F N1(C(c2c(CC)csc2)=O)CC(CNC(c2cc(C(N)=O)cs2)=O)OC(C)(C)C1 C(CC(=O)NC1CCC(C)(C)C1)(C(C)(C)C)NC(Cc1nc(C)sc1)=O C(=O)(CN=c1[nH]c(C)cs1)NC1(CN(C(c2n(CC=C)ccc2)=O)C)CC1 C12(C(=O)NC(CC(C)C)C)CC(CO1)N(C(C1CC(C(C)C)C1)=O)C2 C1(NC(c2nc(C)oc2)=O)CCCCC12CCN(C(=O)CNC(N)=O)C2 c1(C(=O)NC2C(NC(c3c(C)cn(C)c3)=O)CCOC2)cc2scnc2[nH]1 C1(C)(NC(C(CCSCC)N2CCC(NC(=O)OC(C)(C)C)C2)=O)CCCCC1O c1(C2CC(NC3C(C)N(C(=O)OC(C)(C)C)CCC3)C2)cnc2n1CCOC2 c1(C(C(=O)NC2CC(CCNC(CCCC)=O)C2)C)ccc(CC(C)C)cc1 c1(C(N2CC3C(C(=O)NC(c4nccs4)C)(C3)C2)=O)cc2cccnc2[nH]1 Cc1ccc(-n2ncc(C(=O)NC(C)CN3CCCC(C)C3)c2C(C)C)cc1 Cc1cccc(C(=O)NCCCCc2cn(CCCCOC3CCC3)nn2)n1 N1(C(c2c(OC)csc2)=O)CC(C)N(C(c2csc(F)c2)=O)C(C)C1 N1(C(c2c(CC)nc[nH]2)=O)CCC2(CCCC2NC(=O)CC2(N(C)C)COC2)C1 C1(SC)CN(C(=O)CCc2cc(Cl)no2)CC1NC(C1(C)CCCO1)=O C(C(O)CN=c1cc(Cl)nc(CS(C)(=O)=O)[nH]1)NC(C(C1CCC(=O)N1)C)=O N1(C(c2c(COC)cco2)=O)CCN(C(=O)C=C2CCOCC2)CC(CO)C1 CC1=NOC(C(=O)NCCCC2CCCN2C(c2ccccn2)=O)C1 c1(SCCCCNS(CC2(C)N=N2)(=O)=O)csc2cccc(Cl)c12 C1(CCNC(CCSCCC)=O)CN(C(c2cnn(C)c2OC)=O)CCO1 C1(CN(C(COC(CC)CC)=O)C)CCN(C(=O)COC2CCCCC2)C1 C#CC1CN(C(=O)C(C)(F)F)CCN1C(c1ncc[nH]c1=O)=O Cc1c(NC(=O)CCCNC(=O)Cc2cnnn2C)cccc1Cl C(CCC1CC1)(C(=O)NCCN1CCNC1=O)NC(c1cccnn1)=O c1(-c2nc(CCC)nn2CCOCC(F)(F)F)cc2ncccc2s1 c1(C(N2C(C)CC(CNC(=O)CN(C)S(N)(=O)=O)C2)=O)cc2cnn(C)c2s1 c1(CC)cc(C(=O)N(CC(=O)NC(CO)C(=O)OC)CC(C)C)n(C)n1 C(c1ccc(F)nc1)=CC(=O)NC1CC(CNC(=O)CNC(=O)C2CC2)C1 CCCCCCC(C(=O)N1CC(NC(c2cncc(C)n2)=O)C(O)C1)NC(C)=O CC1CCC(F)(C(=O)NCC2(F)CC(CNC(=O)CCS(C)(=O)=O)C2)CC1 c1(C(=O)NCCc2cnc(NCc3ncc(C)cn3)s2)cc(C)cc(Br)c1 c1(C(N(C2CCN(C(C(CCC)CCC)=O)CC2)C)=O)cc2oc(C)c(C)c2[nH]1 N1(C(CSSC)=O)CC(NC(C2CCCNS2(=O)=O)=O)CC12CCOCC2 c1(NC2CC(C)OC(C)C2)nccc(=NCCc2nnc(Br)n2C)[nH]1 c1(CC(=O)NC2CN(C(CNS(NC)(=O)=O)=O)C(CO)C2)ccnc(Cl)c1F c1(C(N2C(C(N3CCC(CC)(CC)CC3)=O)CC(C)CC2)=O)cc2cccnc2[nH]1 C1(C(=O)NCc2c(C)nn(C)c2)CCCN(Cc2ccc(Cl)nc2)CC1 c1(C(=O)OC)cc(CNC(c2cc(C)ns2)=O)ccc1Cl c1(CC(N2CC(C)(NC(CC3N(CC)C(=O)CC3)=O)C2)=O)cnn2c1CCCC2 C(=O)(CC(C)(C)CC=C)NCC(CNC(Cc1ccc(C#C)cc1)=O)CO C1(NC(c2ccccc2C(F)(F)F)=O)CCCN(C(=O)CN2CCOC2=O)CC1 CC1CCC=C1C(=O)NC(C(=O)NCCC1CC=CCC1)C1(O)CCC1 c1(CC2N(c3n(CC)c(C4CC(O)C4)nn3)CCC2)cc(C#N)ccn1 c1(C(=O)NCC(CCNC(C2CN(S(CC)(=O)=O)C2)=O)O)cnn(C)c1C(F)F C(CCC(C)CC(=O)N1CC2CCC(NC(c3coc(C#N)c3)=O)(C2)C1)=C(C)C C(N=c1cc[nH]c2ccc(I)cc12)c1cccc([N+](=O)[O-])c1 c1(C(=O)O)ccc2nc(-c3cn[nH]c3)sc2c1.c1(N2CC2=O)cc2cnc(Cl)cc2s1 c1(C2C(C(N3CCC(O)C(NCC45CSCC4C5)C3)=O)C2)nc2ccccc2[nH]1 C1(N2CC(NC(=O)C(c3cccnc3)NCC3CC3)C2)CCCCCC1O c1(C2(C)CC2)cccc(C(=O)NCC2CCCN(C(C3(Cl)CC3(F)F)=O)C2)c1 CC1(C)OCCC1n1nc(-c2cncc(F)c2)nc1COc1ccc(Cl)cc1 C1(n2cc(CC3N(CC)CCC3)nn2)CCCN(C(=O)Cn2cccc2)C1 c1(C(=O)NCC2(CN(C(=O)C(C)(C)n3cccn3)C)CC2)ccc(C2CC2)nc1 C1(CNC(C(CC)C)=O)CC2(CO1)CN(C(=O)C=Cc1cc(C(=O)OC)co1)C2 N1(C(c2cnc(C)n2C)=O)CCC(O)(CN(C(=O)C2=CCCC2)C)CC1 c1(C(COCC(=O)NC2CN(C(=O)C(O)C3CCCC3)C2)F)ccccc1 C1(F)(C(=O)Nc2c(C)n[nH]c2)CCN(C(c2ccc(N(C)C)cc2)=O)C1 C(=O)(C(CC)(CO)OC)N1CC(CCC)C(C(=O)NCC(c2ccncc2)C)C1 c1(C(=O)NCC=CCC(=O)NCC(CCC)C)c(C)nsc1C C=CCCC(C)N=c1nc(N2CCN(C)C3(CCC3)C2)c2ncccc2[nH]1 O=S1(=O)CC2CC2(c2nc(-c3coc(C4CC4)n3)no2)C1 CC1CN(C(C2CN(C(C3(C#N)CC3(C)C)=O)CC(C)(C)C2)=O)Cc2nncn21 O=C(C1CCCc2nn[nH]c21)NCC(O)CNC(C1CCCSS1)=O N1(C(=O)NC2CC(C)(NC(=O)OC(C)(C)C)C2)CC(C)OC2(CCOC2C)C1 Cc1ccc2c(C(=O)NCCCN(C)C(c3cnn(CC(F)F)c3)=O)coc2c1 Cc1sc(-c2cccs2)nc1C(=O)NCC(C1CCCCN1C)(C)C c1(C2(NC(C3C=CC(NC(c4cc(Br)c(Br)s4)=O)C3)=O)CC2)cccc(Cl)c1 Cc1c(Cl)ccc(C(N2CC3C(C2)N3C(c2ccnc(F)c2C)=O)=O)c1F CCCCC(CC)C(=O)N1CCCC(NC(c2cccc(C(N)=O)c2)=O)CCC1 N1(C(C2CCN(C(C(C)N3CCCC3)=O)CC2)=O)CC2CC3CC2C1C3 n1(CC(=O)NC(CNC(c2cnc(O)s2)=O)C2CC2)cnnc1O CCCC(C)(O)C(=O)N(CCCNC(=O)C(C)CSC)C c1(C(N2CCCC(NC(c3cc(C)sc3)=O)C2C)=O)cc(=O)c2ccccc2[nH]1 CC(C)CC(C(=O)NOCC(C(=O)C(C1CCCCC1)O)=O)N(C)C(C)C O(P(C)(=O)CNC(=O)CC1CC(C)N(C(=O)Cc2cn(C)cn2)C1)CC CC1CCC(CNC(c2cc(C3CC3)no2)=O)CN1C(c1c[nH]nc1Br)=O c1(C(=O)OC)nc(=NCC2CN(C(=O)C3=CCCC(C)(C)C3)C2)c(F)c(Cl)[nH]1 c1(C(=O)NCCCC(C)NC(c2c(OC)cccc2)=O)csc2cc(C)ccc12 c1(C(N2CC3C(CNC(C(C=C)O)=O)(C3)C2)=O)ccc2c(c1)C(=O)NCC2 c1(C(c2n(CC=C)nnn2)NCc2sc(C)nc2C)cc(F)cc(F)c1 CC(F)(F)CCC(=O)N1CCC1CNC(C1(CCS(N)(=O)=O)CCC1)=O c1(C(N(CCCCC(=O)Nc2c(C)csc2)C)=O)cc(F)ccc1C C(=O)(CCS(=O)(=O)C1CCCC1)NC1CCCN(C(C2(C)CC(C#N)C2)=O)C1 CN1CCC(CC(N2CCCCC2CCN(C)C(C2CC3(CSC3)C2)=O)=O)C1=O n1(CCC)nc(C)cc1NC(=O)CN(C)Cc1ccoc1 C(CNC(C1C2CC3C(C2)C13)=O)(CC(F)(F)F)NC(CCC=CC)=O C(=O)(C(CCC(C)C)NC(=O)CCC1CCOC1)N1C(CCCC)CCC1 c1(CNC(c2nnc(Sc3nnnn3-c3ccccc3)s2)C)cc(Br)ncc1F c1(C(=O)NCC(CNC(C(c2ccccc2)N(C)C)=O)(C)O)cc(O)nc(Cl)c1 c1(C(N2CC(CNC(CCCC(C)(C)C)=O)OCC2)=O)nc2ccc(Cl)nn2n1 C(C)(C)(CCN=c1cc(C(C)(C)C)nc[nH]1)NC(Cc1c(C)non1)=O Cc1cn(C(C)(C)C(=O)NCCCN(C(C2CCC(=O)N2)=O)C2CC2)cn1 c1(C(N(C2CCN(C(CN(C(C(C)C)=O)C)=O)CC2)C)=O)cncc2[nH]ccc12 C(C(F)(C(=O)NCC1(C(=O)OC)CCCC1)C(C)C)NC(COCCCC)=O C1(NC(=O)CCn2cnnn2)CN(C(C2CC(F)C2)=O)CC12CCS(=O)(=O)CC2 C(=O)(CC(C)CCC=C(C)C)NC(CC)(C)CNC(c1cncc(SC)c1)=O C(CCC(C)NC(c1nscc1Br)=O)NC(C1C(CC(C)C)C1)=O C1(NC(C2(C(C)(F)F)CC2)=O)CC2CCC(C1)N2C(C1(F)CC=CCC1)=O c1(C(=O)NC2CC(CNC(C3CC(CC)OCC3)=O)C2)ccc2nnn(C)c2c1 CC1CN(C(C2CCCOC2C)=O)CCC1CNC(C12COC(CCO1)C2)=O C1(NC(c2c(CC)nns2)=O)CC(F)CN(C(c2cc3n(n2)CCO3)=O)C1 c1(C(N(CC(CN(C(c2c(C)nns2)=O)C)O)C)=O)cccc(F)c1C c12cc(on1)C(=O)N(CC(O)CO)C2.CC(C(=O)NC1CCCO1)n1cccc1 Nc1c(C(=O)NCC2CN(C(c3ccnn3CCF)=O)CCCO2)cccc1Cl C1(NC(C(C(C)NC(c2n[nH]c(C)c2C)=O)(C)C)=O)CC2CC1OC(=O)N2 N1(C(C2(OCC)CCOC2)=O)CC2CC1C2CNC(=O)CC1(CC)CCOCC1 C1(CNC(c2c(C)nc(C)o2)=O)CN(C(c2ccnnc2)=O)CC(C)(C)O1 CC(C)CCN=C(NCC(c1cccc(F)c1)C)NC1CC1C(N)=O c1(CC(=O)NC2C(CNC(=O)Cc3sccc3Cl)C2)cc(F)ccc1C(F)(F)F c1(C(N(CCCCN(C(CCOCCC)=O)C)C)=O)cnc(C(C)C)o1 C(=O)(C(F)CC(C)(C)C)NCCOCCCNC(Cc1ccc(C)nc1)=O C1(NC(=O)NC)CCN(C(C2(CNC(=O)CC3(C)OCCO3)CCCO2)=O)C1 N1(CCNC(C(C2CC2)NC(C2C(C)(C)C2)=O)=O)CCCCCC1 c1(N2CCC(CC=C)(NC(=O)CCSc3ccccc3)C2)ccnc2ccnn12 c1(NC(=O)CC2CCC(NC(c3cc(F)cc(F)c3)=O)CC2)cccc(Cl)c1Br Cc1cc(C)c(C(N2CCC(CF)(NC(=O)CCc3cnc(C)s3)C2)=O)c(O)n1 C1(CCC)CN(C(=O)C=CCCC=C(C)C)CC1NC(C1(CO)CC(F)(F)C1)=O Cc1ccc(C(=O)NC(CNC(=O)C(C)C(C)C)C(C)(C)C)cc1F c1(C(N2CC(NC(CC3CC(CC)C3)=O)CC2(C)C)=O)cc(C)cc(Cl)c1N CCC(CC(=O)NCCc1ocnc1CNC(c1nsnc1O)=O)C1CCC1 C1(NC(c2cc(C)cc(C)c2O)=O)CCC12CCN(C(C1CC(C)(O)C1)=O)CC2 N1(C(C(C=C)OC)=O)CC2CCC(C1)C(NC(=O)C(C)CC)C2 N1(C(c2n(CCC)ncc2)=O)CC=CC1(C)C(=O)NCCSCC C1(C(C)=O)C(C(=O)N(C2(C(=O)NCCC(F)(F)Cl)CC2)C)C1(C)C N(C1CCc2cccnc21)C(C1OCCC(NC(C2(C)CC2)=O)C1)=O c1(CC(C)NC(=O)CCc2cccs2)nccn1C c1(OC)ccc(C(N2CC(NC(c3cc(C)nnc3O)=O)CC2CO)=O)cc1Cl C(=O)(CCCCC(F)(F)F)NCC1CN(C(C(C)=C2CCCC2)=O)C(C)CC1 Cc1ccc(CCC(=O)NC2CC(C(=O)NCC3(O)CCC3)C2(C)C)cc1 C1(C2C(NC(=O)CC3CC(F)(F)C3)CCO2)CCN(C(c2cnccn2)=O)CC1 C(C(C)C(=O)NC1CCC(CCC(=O)NCCN(C)C)C1)SC C(=O)(CCCCC(C)C)N(CC(CC)NC(c1snc2ccccc12)=O)C C1(CNC(=O)NC2(Cc3ccc(Br)cc3)CCOCC2)CCCC(=O)N1 c1(COCCN(CCC2=CCCCC2)CCOC)nc2ccc([N+](=O)[O-])cc2[nH]1 c1(OCC)cc(C(=O)NC(COC)C(=O)NC2(C(C)C)CCC2)[nH]n1 Cc1cc(COCC(=O)NC2CC(C)(CNC(c3cnc(C)s3)=O)C2)no1 N1(CC(N2CCC(NC(C(C)SCC)=O)C2)=O)CCCS1(=O)=O c1(OC)cc(Cl)c(C(=O)Nc2nc(C(=O)NCc3ccc(F)c(Cl)c3)cs2)cn1 c1(C(=O)NCCCCCNC(CC)=O)ccc(-c2ccc(F)cc2)n1C C(CCNC(=O)C(C)CSC(F)(F)F)(C(C)C)NC(C1(C)CC(=C)C1)=O c1(C(=O)NCCC(C)NC(=O)CCc2ccoc2)cc2c(nc1O)CCN(C)C2 CC1(CNC(=O)COc2cn[nH]c2)CCC(NC(c2ccncn2)=O)C1 C(CC#CC(C)(C)C)NC(C(=O)NCC1CCN(C)C1c1ccccc1)=O N1(C(C2(CC)CC2)=O)CCC2CC2(NC(=O)CCn2c(C)csc2=O)CC1 c1(CC)oc2ccccc2c1C(=O)NC1CCC(NC(=O)CCCNC(N)=O)C1 c1(C(=O)NCCC(C)(C)NC(c2nncs2)=O)ccc(CC2CCC2)cc1 CCC(F)(C(=O)OC)C(=O)NCC(C)(C)Cn1cc(C(O)CC(C)C)nn1 C1(C(C)C)C(NC(=O)CCN2CCN(C)CC2)CCN1C(=O)C=CC1CCOC1 c1(C(=O)NC2COCCN(C(C(C(=O)OC)(C)C)=O)C2)cc2cc(Cl)sc2[nH]1 C1(C(=O)Nc2ccccn2)CC2(C1)CC2F C(c1nccn1CC)=CC(=O)NC(CCNC(C1(CC#C)CCOC1)=O)C C1(OCCN)CCN(C(=O)COC(C(C2ON=C(C)C2)=O)=O)CC1.C1(O)CCOC1 c1(C(=O)NC2C(C)C2)cncc(C(=O)NCc2cccc(O)c2)c1 N1(C(c2cc(CN)c(C(F)(F)F)cc2)=O)CC2CCC1C(O)C2O N1(C(C2(C(N3CCC(C(=O)OC)(OC)C3)=O)CC2)=O)CCC2CCC(OCC)CC12 c1(C(N2CCC(NC(C3CC=CC3)=O)C(F)C2)=O)cc(O)nc2ncccc12 c1(OC)noc(C(=O)NCC2CCCCC2NC(=O)Cc2ccno2)c1Br N1(c2nc(SC)nc(Cl)c2)CCC(C)C(NC(c2cc3cccn3cn2)=O)C1C C(=O)(C(CC)N(C(=O)CC1CC(C)=NO1)C)NC(C#C)CC1CC1 Cc1c(C(=O)N(CCCn2cc(C3CCC3)nn2)C)cnn1-c1ccc(F)cc1 Cc1cc(C(=O)NC2CC(C(=O)N(C(CF)CF)C)C2(C)C)nc(C)n1 C1(C(=O)NCCC(=O)NCC(C)(C)C)CCCC2(CCCCC2)C1 N1(C(C2CCC(CC)O2)=O)CC2CC(C1)C2NC(c1ccccc1C(C)C)=O N1(C(c2ccnc(OC)n2)=O)CC(F)(F)CC1CCNC(=O)C=CC(C)C C(N=c1c(C#N)c[nH]c2c(C)cccc12)C1(NC(CC(CCOC)(C)C)=O)CC1 C1(NC(C=Cc2ccc(SC)s2)=O)CC(NC(=O)CCC(C)(C)F)C12CCC2 Cc1cc(C(=O)NCC(C)(C)NC(=O)CC2C(C)C2(F)F)ccc1OC(F)(F)F N1(C(C2(C)CC=CC2)=O)CC2CCC1C(CNC(=O)CC1CCC3CC13)C2 C1(C(=O)NCC(CNC(c2cn(CCC)nn2)=O)(C)O)CCc2c[nH]nc2C1 N1(C(C=CC=CC)=O)CC(C(=O)N(C)CC2CCOC2C)CCC1C c1(OC)c(C(N2CCCC2C(C)NC(=O)CC2CC(OC)C2)=O)cccc1C c1(CC(C(=O)NC2(C(O)CO)CC2)NC(C(C)SC(C)C)=O)ccc(Cl)cc1Cl C(c1cnc[nH]1)=CC(=O)NCC(C)CNC(C1CC(F)(CO)C1)=O N1(C(C2C(OC)CCC2)=O)Cc2cccc(CNC(=O)C(C)(C)C3CC3)c2C1 c12cc(ccc1N)COC(CC)CNC2=O.C(=O)(CCOC)NCCNC(C)=O c1(C(=O)NCC2C3CN(C(c4n(C)c(Cl)c(Cl)c4)=O)CC32)ccnc2[nH]cnc12 C12CN(CC1N(C)C)C2=O.C(C(C)n1cncn1)OC C1(COC)CN(C(=O)C(O)CC(F)F)CCN1C(c1scc(OC)c1OC)=O c1(C(=O)NCCCS(N)(=O)=O)cnc2ccc(-c3ccc(CO)c(F)c3F)cn12 C(=O)(CCC(C)(F)F)NC1(CF)CCN(C(C(c2cccs2)SC)=O)C1 c1(NC(C2(CC)CN(C(C3CC3C)=O)C2)=O)ccc(CCF)cc1 Cc1c(C(=O)NCC(C)CNC(C2CCCC(F)(F)C2)=O)cc(N)cc1O c1(N2CCC(CC=C)(NC(=O)C=C(C)C(C)C)C2)cnc(C#N)cn1 Cc1n[nH]c(C)c1CC(=O)N(C1CCC(CNC(c2nnn(C)c2C)=O)CC1)C C1(NC(c2cnn(C3CCC3)c2)=O)CC(O)CN(C(c2cc(Cl)ccc2Cl)=O)C1 N1(C(C(c2ccco2)NC(CN(C(=O)OCC)C)=O)=O)CCC(CO)C(C)C1 CC1CCC(Cl)=C(C(=O)NC(C)CNC(c2cc(C(C)(C)C)nn2C)=O)C1 c1(C(CC)N(C(CCOCC#C)=O)CC)ccc(OCCC(=O)NC)nc1 Cc1cc(Cl)c(C(N2CCC(CNC(c3c(C)csc3Cl)=O)C2(C)C)=O)cc1N C1(CC=C)(C(N2CC(OC)CC2CF)=O)CCN(C(c2coc(COC)n2)=O)C1 Cc1cc(N2CCC(C(N3CCC3)=O)CC2)nc(=NCCC2CCC2)[nH]1 c1(C(=O)NC(CNC(c2c(CC)c[nH]n2)=O)CO)cc(C#N)ccc1Cl c1(CCC(=O)NC(C(C)NC(c2cc(COC)oc2C)=O)C)c(C)nn(C)c1C CCCCCCCCC(C)C(=O)NC1CC(NC(c2ccc(C(C)F)cc2)=O)C1 N1(C(c2ccc(F)cc2)=O)CCC2C(CCCN2Cc2ccccc2)C1 CC1CCC(O)(C(=O)NC2CCCN(C(c3ccn(CO)c(=O)c3)=O)C2C)CC1 CC#CCC(C(=O)NCC1CCCC1CF)NC(c1csc(C#N)c1)=O C(C(CO)C(F)(F)F)NC(c1cc(CNC(c2ccc(OC)o2)=O)on1)=O C1(OC)CN(C)C(C)(C(=O)NCCCC(C)NC(=O)C(N2C(C)CCC2C)C)C1 C(c1c(F)cccc1F)=CC(N1CCC(C(C)NC(c2ccnc(S)c2)=O)C1)=O Cc1ccn2cnc(C(N3CCCCC3CN=c3nc[nH]cc3C#N)=O)c2c1 c1(C(N(CC(C)NC(C2CCC3CCC2O3)=O)C)=O)cn(C)c(=O)n(C)c1=O c1(C(=O)NCCC#N)cnc2n1CCN(C(=O)CC1CCCCO1)C2 Cn1nc(CNC(=O)C(F)OC(F)(F)F)cc1C(=O)NCC(C1CC1)C1CC1 CC1CCc2[nH]c(=NCC3CCCC(C)(C)O3)[nH]c(=NCC#CC3CC3)c2C1 C1(NC(=O)CCCn2ccnc2)CC2(C1)CN(C(c1cc(F)cnc1O)=O)C2 C1(NC(CCC=CC)=O)CC2CC(NC(c3cc(C)cnc3C)=O)C2C1 c1(C(C)NC(c2csc(F)c2)=O)cccc(CNC(C2CNC(=O)C2)=O)c1 CCCCC#CC(C)(C)NC(C1(CNC(=O)C(C)(C)C(C)O)CCCC1)=O c1(Nc2cc(NCC3(C(C)C)CCCC3)ncn2)ccc2sccc2c1 c1(OC)cc(F)ccc1S(=O)(=O)NC(Cc1ccc(C#N)cc1)C(=O)O c1(C(N(CCCNC(C2COC(=O)C2)=O)C)=O)[nH]nc2c1COC2(C)C c1(OC)ccc(C(=O)NC2CCCCN(C(C3CN(C)C3)=O)C2)cc1S(C)(=O)=O c1(C(=O)NCC2N(C(C(C)OCC)=O)CCCC2)cc(O)ccc1Br C1(CCC(=O)NCC23CC2CCN3C(=O)CC(F)(F)Cl)CCC(O)CC1 c1(C(N2CCC(CN(C(=O)CC3CCC(O)C3)C)CC2)=O)cc2n(n1)CCOC2 CC(C)(CCCNC(=O)CSc1ccccc1Cl)NC(=O)CCC1CCC1 c1(C(N(CCC(C)NC(C2(C=C)CC2)=O)C)=O)ccc(NS(C)(=O)=O)cc1Cl CCC(C(=O)NC(c1ccccc1)C(C)NC(c1csnc1OC)=O)NC(C)=O C1(C2CN(C(C3CCOC3)=O)C2)(NC(CCCOCCOC)=O)CC1 CCC(CC)C(=O)NCC(=O)NCC(CC1(NC(=O)COC(C)C)CC1)=O C(C)(C(C)NC(C1(F)CN(C(C2CCC2C#N)=O)C1)=O)(C1CC1)OC CCCCC(=O)C(=O)NC1CC(O)CN(C(=O)CC2(COC)CC2)C1 c1(C(=O)NCCN(C(CCOC)=O)CC(C)O)ccnc(C)c1O c1(C(=O)NC2(C(N3CC(N(CCOC)CC)C3)=O)CC2)cc(C)sc1N N1(C(CN(C)CCO)=O)CCCC2C1CCCN2C(c1c[nH]nc1C(F)(F)F)=O C1(C(N2CC(O)(CNC(=O)CNC(C3CCC3)=O)C2)=O)CCn2ccnc2C1 c1(CCC(N2CCN(C(=O)CC3(CO)CC3)C3CC23)=O)c(Cl)cccc1Cl C1(N(C(C(CCC)NC(=O)Cc2ccccc2O)=O)C)CCN(OC)CC1 C1(C(=O)NC2C(CN(C)C)C2)CCN(C(C2CC(F)C2)=O)C1(C)C CC(=O)CCCC(C)C(=O)NC(C)(C)CCCNC(C1CCn2cnnc2C1)=O Cc1ccc(-n2nc(-c3ccc(F)cc3)nc2-c2cnn(C)c2O)cc1 N1(C(Cc2c(C)noc2)=O)CC2CCCC1C2CNC(c1ccc(CF)cc1)=O CC1(C)CC(NC(=O)CCc2ccco2)CN(C(=O)CC2(C)CCS(=O)(=O)N2)C1 N1(C(c2cc(C)[nH]n2)=O)CCC(C)(CNC(=O)CCC2CCCCC2)C1 c1(N(C)CC2(CN(C)C)CCCCC2)ccncc1S(=O)(=O)N1CCC(F)CC1 O=C(CS(=O)(=O)CCCc1ccccc1)NC1CC2CC1N(C(=O)CCF)C2 C1(CC(=O)NC(C)C=CC(=O)N(C2(C)CC2)C)CCOC1 C1(NC(CNC(C2N(C(CN3C(C)CCC3)=O)CCC2)=O)=O)CCS(=O)(=O)C1 C(C(=O)NCC1(C(=O)N(CC(C)C)CCOC)CCCO1)(C(C)C)OC C1(N)(C(=O)O)CCN(C(=O)C(c2csc(C(F)(F)F)c2)C2CC2)CC1 C1(NCc2cc(C)oc2C)CC2CCC1CC2 C(C(C(C)(C)C)NC(C1(C2CCCO2)CC1)=O)NC(C(C)Cc1cnc[nH]1)=O C(=O)(CCC(=O)NCCN1CCC(N(C)C)CC1)NC(C1C(C)(CC)C1)=O N1(C(C2C(CCOC)C2)=O)CCC2CN(C(=O)CCc3ncccc3C)CC2C1 C(C(O)CC(=O)N(C)CC1(O)CCCC1)NC(c1cc(C)[nH]n1)=O c1(C(N2CC(NC(c3nccc(C(C)(C)C)c3)=O)C3C2C3)=O)cc(F)ccc1F C(CN=C(NC1CC(F)C1)N1CCC(C2CC2)CC1)OC(F)F N1(C(C2C(C)C2)=O)CC2(C1)SCCC2NC(=O)CC1NC(=O)NC1=O c1(-n2cc(C(C)NC(=O)C(F)(F)c3csc(C(F)(F)F)n3)nn2)cc(F)ccc1F c1(C(=O)NC2CCC2NC(c2n[nH]c3c2CCC3)=O)cc([N+](=O)[O-])cnc1O C(=O)(C1=CCCC1(C)C)Nc1cccc(NC(c2cnn(C)c2N)=O)c1 c1(C(N(C(C)C)CCNC(=O)C(F)(F)c2nccs2)=O)cnc2n1CC(C)CC2 C1(CCOC)CN(C(c2sc(=N)[nH]c2C)=O)CCN1C(c1cnn(C)c(=O)c1)=O n1(CC(=O)N(CCOC2CCCCC2)CC)ncc(Br)n1 C1(NC(C2C(C)CCN2C(=O)CCCCC2CC2)=O)CC2CC1CC21CC1 CCCC(CC(C)C)C(=O)NCCNC(c1nnn(C)c1CC)=O CCC(C)(C#N)C(=O)N1CC2CC1CN2C(=O)Cc1cc(C(C)C)no1 N1(C(c2cc(C)no2)=O)CC(F)CC1CNC(=O)C(C)c1ccon1 c1(C(=O)NCCOCCCNC(C2OCC(C)(C)C2)=O)cccn2c(O)nnc12 c1(N2CCC(C(=O)NC)CC2)nc(N2CCC(F)(F)C(CO)C2)c2c(n1)CSC2 N1(C(c2c(CC)cco2)=O)CC2CN(C(C34CCC(F)(CC3)CC4)=O)CC2(C)C1 C1(c2n(C)ccn2)CS(=O)(=O)CCO1.C1(C)(C(=O)O)Cn2nnc(n2)S1 N1(C(c2cn(CCC)nc2)=O)CCC(CO)(CNC(=O)CC2(OC)CC2)C1 c1(C(=O)NC2C(Nc3ncc(OC)cn3)CCCC2)c(C)c(C)c(C)c(C)c1C c1(C(=O)NCC(CC)NC(=O)CC(C)(C)COC(C)=O)c(S(C)(=O)=O)cnn1C CCC(O)C(F)(F)C(=O)N1C2CCC1CN(C(c1cccc(SC)c1)=O)C2 C(=O)(CCCC(=O)NCC)NC1CC(CNC(COCC=C)=O)C1(C)C Fc1ccc(COCC2CCN(Cc3cc(C4CC4)on3)C2)cc1 c1(C(N2CC(C)N(C(=O)CC3CCCCO3)CC2)=O)cn2c(n1)C(=O)N(C)CC2 C1(NC(CCC=C)=O)COCCC1NC(c1ccnn1-c1ccccc1)=O C(C(=O)N1CC(C)(O)CO1)C1(N(C(=O)CN2C(=O)CNC2=O)C)CC1 c1(C(=O)NC(CN(C(c2c(OC)ccc(C)c2)=O)C)C)c(C)cc(O)cc1C C=CCCCC(=O)N1CCC(CN(C)C(c2ccc(OC)s2)=O)CC1 N1(C(C2(CC)CC2(F)F)=O)CCC2CN(C(c3cc([N+](=O)[O-])nn3C)=O)CC2C1 c1(OCC(N2CCCCC2)=O)nccc(NC2CC(Cl)=NO2)n1 N1(C(C2(C)CC3(CCC3)C2)=O)CCOC2(CCCN(C(C3(O)CCOC3)=O)C2)C1 c1(C2C(C(=O)OC)C2)cc(CNC(=O)NC23CCC(C(C)(C)C)(C2)C3)c(C)o1 C1(N(C(=O)CSc2nncn2C2CC2)CC)CCCN(C(=O)C(C)SC)C1 Cc1ccc(-c2nc(C(=O)N(CCN(C)C(c3n[nH]cc3Cl)=O)C(C)C)cs2)o1 C1(C(C)C)SC(=NCC(C)SC(C)(C)C)N(C2CCNC(=O)C2)C1=O c1(OC)ccc(Br)c(F)c1NC(=O)CN1CCC(c2ccc(NC(C)=O)cc2)C1 N1(C(=O)CC(O)C2CC2)CC2(C1)CN(C(C1CCC3(CCC3)CC1)=O)CC2CO C(=O)(C1CCCc2cncn21)N1C(CN(C)C(c2cccc[n+]2[O-])=O)COCC1 c1(SC(CC(=O)NCCN(CCC)C(C2CCC2)=O)C)nn(C)c(C2CC2)c1C C(CC(O)CC(=O)NC1CC12CCCC2)SC C1(NC(c2c(OC)nn(C)c2)=O)COCCN(C(=O)CC2C=CCCC2)C1 N1(C(C(C2CCOCC2)C)=O)CC(C)(C)CC1C(=O)NCC(C)N(C)C c1(C(=O)NCC2CCN(C(c3c(C)ncnc3)=O)C2)nc(C(F)(F)F)ccc1N CCCCCCC(C)C(=O)NCC1CCN1C(=O)CCSCC C1(O)(C(N(CCCCCCNC(c2ccc(Cl)o2)=O)C)=O)CCC(C)(C)CC1 N1(C(C=C(C)C2CC2)=O)CC(C)CN(C(c2ccnn3ccnc23)=O)C(C)C1 C1(C(=O)NCC(C(C)C)OC)(NC(C2C=C(C)CS2)=O)CCN(C)C1 Cc1nc2cncc(C(N3CCC(N(C)C(c4cc(Cl)ns4)=O)C3)=O)c2[nH]1 N1(C(C2(C)CC2(Cl)Cl)=O)CCC2CN(C(=O)C=Cc3cnc[nH]3)C2C1 C1(C2CCC2)(CNC(C=CCC)=O)CCN(C(=O)C(C)CCCOC)CC1 C(CC(O)C(=O)NC1CC(C)(NC(C2CC(C)(O)C2)=O)C1)SC C(CNC(=O)C(C(C)C)SC)(C(C)(C)C)NC(C1CC(CC)(CC)C1)=O c1(-n2c(CCC(C)(C)F)nc(C(CC)O)n2)cccc2ncccc12 N1(C(c2ccc(C(C)(C)C)cn2)=O)CC2(CCC2)C2COCC12 C1(C)(C(N2C(CC)C=CC2)=O)CC12CCN(CC1CCOC1)CC2 Cc1noc(C)c1C(=O)NCC(=O)N(CC(O)CNC(=O)C(=O)NCC1CC1)C C1(C(OC)NC(=O)C(C)Nc2cccs2)C2CN(C(=O)CC3(C)CCOC3)CC12 Cc1nc(O)[nH]c1C(=O)NC1(CN(C(=O)C(O)CC2CCCC2)C)CC1 Cc1nc(C(C)C)oc1C(=O)NCC(C)NC(c1cnc(-c2ccc(Cl)cc2)s1)=O c1(CNC2C(C(=O)Nc3c(C(=O)OCC)c(C)sc3)CCC2)ccc(F)cc1I c1(CC(=O)NC(C)CNC(c2c[nH]c(=O)cn2)=O)ncn2c1COCC2 C(=O)(C(C)CC(F)F)N(C1CCN(C(C2(COC)CCC2)=O)C1)CC#C c1(C(N2CC3CCN(C(c4cc(Br)ncc4F)=O)C3C2)=O)cc2cnccc2[nH]1 C(=O)(CCCC(=O)N1CCC(C(C)(C)CNC(=O)Cc2ccon2)CC1)OCC c1(CC)cc(C(N2CCC(NC(=O)C=C3CCC(C)C3)C(F)C2)=O)ccc1O C1(CCCCC)CCC(C(=O)N(C)CCOCCN(C)C(c2ccnn2C)=O)O1 c1(CSC)ccc(C=CC(=O)NCC(C2CCC2)NC(C2(CO)CC2)=O)cc1 CCC(CNC(=O)C(F)C1CCC1)(CC)Nc1nnc(C)o1 CC1CC=C(C(=O)NCC2(CCNC(C3CC34CCOC4)=O)CC2)CC1 C1(NC(CN(C)C)=O)CCC12CN(C(=O)CCc1cccc(F)c1F)C2 C(C(C)(C)CS(=O)(=O)NCC1CNC(C)(C)C1)OC C1(C)(NC(CCOC)=O)CCCN(C(=O)CCc2c(F)cccc2F)C1 C=C(C)CN=C(NCC1(C#N)CCCC1)NC1CC(OC)C12CCC2 c1(C(=O)NCC(CC(C)C)NC(C2Cc3nccn3C2)=O)cc2ncccn2n1 CCC(C)(C(=O)N1CCN(C(c2ccc(C(C)C)c(F)c2)=O)C2(CC2)C1)C(F)F C1(CNC(c2c(CC)occ2C)=O)CCN(C(=O)CSC)C12CCC2 Cc1ncn(-c2ccc(NCc3c(Br)cnn3C(C)C)cc2)c1C C1(C)(SC)CCN(C(C2CCN(C3CNC3)CC2)c2cn(CCO)nn2)C1 c1(C(=O)NCC2C(C)CN(C(=O)CNC(=O)C(C)(C)C)C2)nc2c(s1)CCCC2 N1(C(CC2OCCN(C(CC=CCC)=O)C2)=O)CCC(F)(C#N)C1 n1(CC(C)O)cc(-c2nc(CCC(C)(C)C)nn2CC(N)=O)ccc1=O c1(C(C)=O)cc(C(=O)N(C)CCNC(C2CCC3C2C3(F)F)=O)ccc1O N1(C(C=CC)=O)CCCCC2(C1)CN(C(c1cccc(C(=O)OCC)c1)=O)C2 N1(C(C2(OC)CCOCC2)=O)CCN(C(=O)C(C)SC)C(C2CCC2)C1 c1(C(N2CC(CNC(C3C(C)OCCC3)=O)OCC2)=O)ccc2c(c1)nnn2C c1(CC(C)C)oncc1C(N1CCC(N(CCO)C(C2CCCCO2)=O)C1)=O c1(-c2nnc(N(CC#C)C)n2CC2CCCNC2=O)ccc(F)c(OCC)n1 c1(C(c2nnnn2C(C)(C)C)NC(CC=C)CC)nc(Br)c2ccccn12 C1(CC)CC(C)CN(C(=NCCC(C)(C)S(C)(=O)=O)NCc2ccco2)C1 c1(CNC(C2(COC)C=CCN2)=O)cccnc1O N1(C(COC)=O)CCN(C(c2cnn(CCO)c2)=O)C2CCCC2(C)C1 C1(C(=O)NCCCOCCCNC(c2ccn(CC)n2)=O)CC2CCCCN2C1 Cc1nsc(CNCC2(CSC)CCN2C(=O)OC(C)(C)C)n1 CC1(C(N2CCOC(CNC(c3ccncc3C(F)(F)F)=O)C2)=O)CNC(=O)C1 CN1CC(NC(c2ccc(CNC(=O)CC3CC4(CC4)CO3)o2)=O)C(F)(F)C1 Cc1ccc(C(N2CCC(CN(C)C(c3ccc(C4CCOC4)s3)=O)C2)=O)cc1 c1(OC)cccc2cc(C(=O)NC3CC3NC(c3cnc(C)[nH]c3=N)=O)oc12 N1(C(c2cc(CCNC(C3(C)C(CC)CCC3)=O)on2)=O)CCc2nocc2C1 c1(C(=O)NCCC(C)NC(C2N(CC)CC2)=O)ccc(F)c2ccncc12 CC(C)CC(C)(CNC(C1CS(=O)C1)=O)NC(=O)CC1CC(F)(F)C1 CCC(C)C(O)C(C)C(=O)N(C1CCN(C(c2cn(C)c(=O)cn2)=O)C1)CC C12CN(C(C)(C)C1)C(=O)C(=O)N1CCC(C1)N2.CC1(CCC2CC2)CC1 c1(C(=O)NC(C2CN(C(=O)Cc3cnco3)CCO2)C)ccc2ccccc2n1 N1(C(C2N(Cc3ccc(OCCC)cc3)CCCC2)=O)CC(C)OCC1C c1(C(N2CCC(CNC(c3ccc(CC)cn3)=O)C2)=O)ccc(Cl)c2occc12 CC1CNCCN1C(=O)C(=O)Nc1cccc(NC(c2ccccc2)=O)c1 C1(C(N2CCC(C3(C)N=N3)C2)=O)C2CC(O)C(C2)N1C(=O)CCc1nncs1 CC(CCNC(=O)CC1(CO)CC1)NC(=O)CCN(S(C)(=O)=O)C Cc1nc(C)c(C(=O)NC2(C)CC(C(N3CC(CO)(CO)C3)=O)C2)s1 C1(NC(CC2(C)N(C(CC3N(C)CC=CC3)=O)CCC2)=O)COC2(CCC2)C1 CCCCC(CCCC)C(=O)N1CC(NC(C2(CO)CCCO2)=O)C(O)C1 c1(C(=O)NCCN(C(C=NOC)=O)C2CC2)cc(S(=O)(=O)N(C)C)oc1C CCCC(C)(O)CC(=O)N1CCN(C(c2nc3cccnc3s2)=O)C(C(C)C)C1 C1(NC(c2n(C)cnc2)=O)CCCN(C(=O)COCCc2cccs2)C1 C1(C(N2CCCC(N(C(=O)CCN3CCCC3)CC)C2)=O)CCn2nnnc2C1 c1(C(=O)NC2C(NC(C(C)(C)OCC)=O)CC(F)(F)C2)ccc2oc(=O)oc2c1 N1(C(c2cnc(CC)s2)=O)CCC2CC2(C(=O)NCC2CC(C#N)C2)CC1 C(C)(C(O)C(=O)NCC(C1CCN(C(=O)CCc2ccn(C)n2)CC1)(C)C)OC N1(C(C2(C(C)C)CC2)=O)CCC(NC(c2ccc3[nH]ccc3n2)=O)C(F)(F)CC1 C(=O)(C1CCCc2[nH]nc(I)c21)N1C(c2cc(C)c(Br)cc2)CCC1 CC(CCCCNC(=O)CCN1CCCCC1=O)NC(=O)Cc1nnc(O)s1 c1(C(N2CCC(NC(C3C(F)(F)C34CC4)=O)C2)=O)[nH]nc2ncnc(O)c12 C1(CN(C(=O)Cc2sccc2Cl)C)CC(F)CN1C(=O)CCc1cnoc1 C1(C(N2CCC(NC(CC(=O)OCC)=O)C2C)=O)CC(C2CCCC2)C1 C12(C(=O)NCCCNC(c3nccnc3-n3ccnc3)=O)CCCCC1CCC2 N1(C(C(C)c2cc[nH]n2)=O)CC(NC(C2CC(F)(F)C2)=O)C(O)C1 N1(CC=C)C(=O)C(=O)N(CC(=O)N(C(C)CNC(c2cc(C)n(C)n2)=O)C)C1=O c1(-c2nc(-c3sc(C)c(Br)c3)on2)ccc([N+](=O)[O-])cc1 c1(OC)cc(NC2(CNC(=O)C=Cc3ccco3)COC2)ccc1[N+](=O)[O-] c1(C(N2CCC(C(C(=O)Nc3c(CC)n[nH]c3)C)C2)=O)cnc(O)c(C)c1 Cc1c(C(N2C3CCC2CN(C(c2ccon2)=O)C3)=O)nc2sccn12 C1(C2CCN(C(c3c(C)c[nH]n3)=O)C2)CCCCN1C(c1coc(C(N)=O)c1)=O N1(C(CSc2nc(C)[nH]n2)=O)CCC(C(C)CNC(c2cscn2)=O)CC1 C1(NC(c2c(C)cno2)=O)CC(CNC(c2cnoc2C)=O)C12CCC2 c1(NC(C2(Cc3nnnn3C3CC(F)(F)C3)CCCC2)=O)cnn(CC(F)F)c1 N1(C(C(C(C)C)SC)=O)CC2(C1)SCCC2NC(c1cccc(C(C)(F)F)n1)=O C(N=c1[nH]c2c(c(=NCCCn3nccn3)[nH]1)CCCCC2)c1c(C)ncs1 c1(CN2C3C(C(=O)Nc4cnc5cc[nH]c5c4)C(C3)C2)cc(F)c(I)c(F)c1 c1(CC(N2CCN(C(c3cn(CC)nc3C)=O)C3C2C3)=O)ccc2ncnn2c1 CCC(C(=O)NCC12CC(CN1C(c1ccc(N(C)C)cc1)=O)C2)C(C)O C1(NC(=O)CCc2cn[nH]c2)CCN(C(C2CCS(=O)(=O)CC2)=O)C12CCCC2 C1(C(N2CC3CN(C(C4(C=C)CC4)=O)CC3(C)C2)=O)CC(c2ccc(F)cc2)=NO1 C=C(CNC(c1cc(C(C)(C)C)c[nH]1)=O)CCNC(c1cc(COC)no1)=O c1(C(=O)OC)sc(Cl)cc1NC(=O)N(CCCC(C)O)C c1(C(=O)NCCOCCCNC(C2CCC3(CC3)C2)=O)noc2c1CCCCC2 C(=O)(C(F)(F)c1ccccc1)NCC1CC(CCN=[N+]=[N-])C1 Cc1cc2c(C(=O)NCC(CO)NC(=O)CSc3cccs3)cccc2[nH]1 C1(NCC(=O)NC2CC2)CCS(=O)(=O)C2(C1)CC(NC(N1CCOCC1)=O)C2 CC12CC(NC(C3CCSCC3)=O)(C1)C1(CN(C(C3(F)CC=CCC3)=O)C1)O2 CC(C)(C)CC(C)(C)C(=O)NCC(CO)NC(=O)C(O)CC1CCCCC1 CC1(CNC(C2CCN(C(=O)OC(C)(C)C)C2)=O)CS(=O)(=O)CCO1 CCCCCCC(=O)N(C1CCN(C(=O)CCc2cccnc2)C1)CC1CC1 C1(NC(c2ccon2)=O)CC2CC1N(C(=O)C=Cc1sccc1Br)C2 C1(O)(C(=O)NCCCN(CCCCNC(CC(C)OC)=O)C)CCC(C)CC1 c1(CC(=O)NCC(O)CNC(c2ncccc2O)=O)ccc2ncccc2c1 c1(C(=O)NC2C(NC(CSCCC(C)C)=O)CCC2)cc(C(F)(F)F)cc(N)c1 N1(C(c2ccc(C(C)C)cc2)=O)CCN(C(c2ccnc(O)c2)=O)C(CC#N)C1 c1(C(C)C)ccc(F)cc1C(=O)NC1(CO)CN(C(c2ccc(=N)[nH]n2)=O)C1 C1(C)(CCNC(CNC(C(CC)C)=O)=O)CCN(C(=O)CSCCC(F)(F)F)C1 C1(NC(=O)CCN2CCC2)CN(C(=O)CCc2ccccc2O)CC1O N1(C(c2nc(C)oc2)=O)CC2C(CNC(=O)CC3CCC(O)C3)C2C1 c1(-c2nc(C3(OCCCOC)CCC3)on2)cc(C2CCCC2)[nH]c1C C1(CNC(CCCC#N)=O)CCCCN(C(C2(n3cncn3)CC2)=O)C1 CC1CN(C(C2(NC(C3CC3C3CCC3)=O)CC2)=O)CCO1 c1(C(=O)NCC(CCCC)NC(=O)Cc2ccoc2C)ccc(Br)nc1N c1(C(N(C)CCOCCN(C(=O)C(O)C2CC2)C)=O)ccc(C(F)(F)CF)cc1 c1(OC(CC)C)cc(CNC(=O)NCC(c2ccc(C)nc2)(C)C)ccn1 CCCC(CC)CCC(=O)NCC=CC(N1CCCN(C=O)CC1)=O Cc1ccc(Cl)cc1NC(=O)C(C)(CO)NC(C1CC(C)(F)C1)=O c1(CC)ccc(N)c(C(=O)NC(C)(C)CNC(c2cc(C)cc(Cl)c2)=O)c1 c1(C(N(CCCNC(c2ccc(C(C)C)o2)=O)C(C)C)=O)cn2ccnc2s1 C(CC(C)C(=O)N1CC2CC2(CNC(c2ccc(NC(C)C)cn2)=O)C1)OC S(=O)(=O)(c1ccc(Br)cc1NCc1cn(C)nc1Br)N1CCCC(C)(OC)C1 CCC(CC(=O)NC(Cc1ccco1)C(=O)N(C(C)CC(F)(F)F)C)SC C(=O)(CC(C)C(F)(F)F)N1CCC(C(=O)NCc2nc[nH]n2)(CC)C1 C(C)(CO)(C(=O)NCC=C1CCN(C(C2C(F)(F)C23CC3)=O)CC1)OC c1(CC(=O)NCC(CCOC)NC(C2C(=C)CC2)=O)cccc(Cl)c1 c1(C(=O)NCCCN(C(C2(CC)CC2)=O)C)ccc2c(n1)CCCC2 C(=O)(NN(C)CC(C)O)NCC1CCC(CCCCC)O1 N1(C(C(COC)N(C)C)=O)CCOCCC1C(=O)Nc1ccc(O)nc1 C1(NC(c2cncnc2)=O)CN(C(c2ccc(CO)cc2)=O)CCC12CCC2 CC1CN(C(c2ccccc2Br)=O)CCCN1C(c1ccn(C2CCC2)n1)=O CCCCCC(C)(C)C(=O)OCC(=O)Nc1cccc(N2NC(=O)CCC2=O)c1 c1(CCC(=O)NCCN(CCOC)C(c2ccc(C)nc2)=O)nnc(C)n1C C1(NC(CCCC)=O)CN(C(c2cc3ccsc3c(O)n2)=O)CC2(CCC2)C1 c1(C(=O)NC(COCC)C(=O)NC2CC2(C)CC)cnn(C)c1Cl Cc1cnnc(O)c1C(=O)NCC=CCNC(=O)C=Cc1cn[nH]c1 N1(C(c2ccncc2)CC)C(=O)NC(C)(c2ccc([N+](=O)[O-])cc2)C1=O C(c1ccsc1C(F)(F)F)=CC(=O)NC(C1CCS(=O)(=O)C1)CO CN1CC(C)(C(N2CCCC2C(=O)NC2CC(O)CC2O)=O)CC1=O c1(C(N(C)CC2(NC(c3ncc(OC)cn3)=O)CC2)=O)c[nH]c2c(F)cccc12 C(N=c1cc[nH]cc1[N+](=O)[O-])C1CN(C(COC(CC)C)=O)CC12CCC2 C(=O)(C(CCC(C)C)N(C)C)NC1C(CNC(C2(SC)COC2)=O)CCCC1 Cc1ncc(C#N)cc1NC(C1CCCCCCN1C(=O)CC1CC1(C)C)=O C1(C(=O)NC(C2(O)CCCC2)C)CN(C(=O)CC2=CCCCC2)CC(C)(C)C1 Cc1cc(Br)c(CC(=O)N(CC(C)N(C)C(c2cnccn2)=O)C)s1 CCC(C)CC(=O)NC1(C(=O)NCC2CCC2NC(=O)OC(C)(C)C)CCC1 C1(COC)CN(C(c2ccn(C)c2)=O)CCN1C(C1COCCC1(F)F)=O c1(C(=O)OC)c(C)nc(CC2CCCN(c3c(C(=O)OCC)cccn3)C2)nc1C C(=O)(CCCCC(C)C)N(CCNC(c1c(C)ccc(NC(C)=O)c1)=O)C1CC1 C1(NC(c2scc(C)c2)=O)CCC2(CCN(C(c3ccc(C#N)o3)=O)CC2)C1 C1(NC(=O)CC2=CCCC2)C2COCC1CN(C(=O)C(F)F)C2 CC12CCCC1N(Cc1cccc(-c3ccc4c(c3)CCC4)c1)CCC2 S(=O)(=O)(c1ccc(=NCCCCn2cnnc2)[nH]c1)NCc1cnn(CC)c1C c1(C(=O)NCC2CCN(Cc3ccc(C)cc3)CC2)cc(Br)cn(CC#N)c1=O C(=O)(C(F)(F)C(F)(F)F)N1CCC(=CCNC(C(C(C)C)OC)=O)CC1 C1(C(=O)NC(c2ccccc2Br)CN)CCC2(CCNCC2)C1 C1(NC(C(=Cc2cccs2)C)=O)CCN(C(=O)C(O)C(C)C)CC12CCC2 c1(NC(C)(C)CCNC(c2ccc(C(N)=O)c(Cl)c2)=O)ncc2cccnc2n1 c1(C(N2CCC(C)(CNC(c3c(C)ccnn3)=O)CC2)=O)cccn2cnnc12 C(=O)(C1=CCCOC1)N1CCN(CCN(C)C(C2(F)CC=CC2)=O)CC1 C#Cc1ccnc(C(=O)NC(CNC(c2ccc(OC)s2)=O)C(C)C(C)C)c1 CC(C(=O)NCC1CCN1C(=O)CC1CNC(=O)O1)S(C)(=O)=O C(=O)(C1=NOC(C)(C)C1)NCC#CCNC(C(=O)Nc1cccc(C)c1)=O C1(C(=O)NCC2(NC(C3C(C)CC3)=O)CC2)CCC(C)(O)CC1 C=C=C(C)CC(=O)NC1CCC(F)(CNC(C2CC(O)(c3ccccc3)C2)=O)C1 CCN=C(NCC1CCCCN1Cc1ccccc1)NCC(C)(F)F C1(c2c(OCC)cccc2OC)NC(=S)N(CC2CC2)C2=C1C(=O)NC21CCC1 N1(C(c2c(CNC(C3(C(C)=O)CC3)=O)noc2)=O)CCCC2CC12 c1(OC(C)C)ccc(CC(N2CCCC2CN(C(=O)C(C)O)C)=O)cc1 C1(NC(c2ccc(C#C)o2)=O)CCCN(C(=O)Cc2csnc2C)CC1 c1(NCCN(c2ccc(Br)cn2)C)ccc([N+](=O)[O-])o1 C1(CNC(c2cc(OC)no2)=O)CCN(C(=O)Cc2ncc(Cl)s2)CC1O C(=O)(Nn1cnnc1C)C1(CC=C)CCN(C(C2COC(=O)N2)=O)C1 c1(C(C)C)ccc(O)cc1C(=O)NC1CN(C(c2occc2F)=O)C1 c1(C(N(C)CC2CCN(C(C=C(C)C(F)F)=O)C2)=O)ccc([N+](=O)[O-])cc1F CC1Cc2c(Br)cccc2CN1C(C1CC(F)C1)=O CCCC(C)(CC)C(=O)NC1CC2(C1)CC(C(=O)Nc1cnccc1C1CC1)C2 N1(C(COCC(C)(C)C)=O)CC2OCC(NC(c3ccc(C(N)=O)cc3)=O)C2C1 C(C)(CCC(=O)N1CC2CC2(NC(=O)CN(C)CCO)C1)OCC C1(C(=O)NCCCCCCN(C)C(C2CN(C3CCC3)C2)=O)CC(C)(C)OC1=O C1(NC(c2ccncc2C(F)(F)F)=O)CCCN(C(C2(Cl)CC2)=O)CC1 C1(NC(CC23CC(C)(OC2)C3)=O)CCCN(C(=O)CC2(O)COC(C)(C)C2)CC1 N1(C(c2cc(CNC(c3cc(C)[nH]n3)=O)sc2)=O)CC(C(C)C)CCC1C C(=O)(CC(C)(C)C(=O)OC(C)(C)C)N(C(C)CNC(=O)CC1(C)CCC1)C N1(C(C2(C)CC3CCC2C3)=O)CC2CCCC(C1)N2C(C1(F)CCC1)=O c1(-c2ccc(OC)nc2)cn2c(n1)CN(C(c1cc(C#N)c(SC)nc1O)=O)CC2 Cc1cc(C(=O)N(C2CCCC(NC(=O)CSC(F)F)C2)C)ccc1C#N Cn1ncc(C(N2CCC(N(CC3CC4CCC3O4)CC3CC3)CC2)=O)c1Cl c1(C(C(=O)N(CC(C)CNC(C2(C(N)=O)CC2)=O)C)O)ccccc1F CCC(C)C(=O)C(=O)N1CCC(O)C(NC(=O)C(C)SC(C)C)C1 c1(C(=O)NC(C(C)NC(=O)CCc2nnnn2C)C)c[nH]c2ccccc2c1=O c1(NCC(=O)NCC2(F)CC(NC(c3c(C)cccn3)=O)C2)ccccc1C#N Cc1cc(CN(C)CC2CN(C(=O)CCOc3ccc(Br)cc3)C2)cc(C)n1 Cc1n[nH]c(C)c1C(=O)NC1CCC1NC(=O)C=C1CCCCC1 N1(CC(C)(C)NC(=O)OC(C)(C)C)CCC(CO)C(Cc2noc(C3CC3)n2)C1 c1(CC)cccc2c(CC(=O)NCCCCNC(=O)C(C)(C)OC(C)C)c[nH]c12 C#CCCN=C(NCCN1CCOCC1)NCc1ccc(Cl)c(F)c1F C1(CC)C(C(N2CCC2)=O)CCCN1C(c1c[nH]c(C(N)=O)c1)=O c1(C(F)F)ncc[nH]c1=NCCc1ccc(F)cc1F c1(CC(=O)NC2(C)CC(CNC(CCCOCCC)=O)C2)cc(F)ccc1F CCS(=O)(=O)c1ccc(-c2cncc(CNc3ncc4ccn(C)c4n3)c2)cc1 N1(C(c2cccc(CC)n2)=O)CC2(C1)SCCC2NC(=O)C=Cc1ccco1 CN=c1nc(N2CCC(NC3CC3)CC2)[nH]c(=NCCP(C)(C)=O)[nH]1 N1(CC)CCN(C(=O)C(F)(F)C2(O)CCC2)CC1.C1(NC(C)=O)CN(C)CC1O N1(C(CCCCCC=C)=O)CC2CCCC(CNC(C3(Cl)CC34CCC4)=O)(C2)C1 N1(C(CSC)=O)CCn2ncc(CNC(c3ccncc3)=O)c2C1 C1(NC(CC2C(C)C2)=O)CC2(CCCN(C(c3ccc(Cl)nc3Cl)=O)C2)C1 c1(-c2ccc(OC)nc2)csc(=Nc2ccccc2)n1CCc1ccn(C)n1 c1(CCC)nnsc1C(=O)NC1(COC)CN(C(=O)C(C)CN(C)C)C1 C(C)(C(C(=O)NC12CCN(CC1)CC2)C(C)C)NC(CCNC(=O)NC)=O c1(C(=O)NCC(C)NC(C2CC2C2CCC2)=O)ccc2c(c1)nc(O)n2C C1(NC(CC(CC)CC)=O)CCC2(CCCN(C(=O)Cc3cnnn3C)C2)C1 CC1OCCC1(F)C(=O)NCC#CCNC(=O)CC1CC1c1cccc(Br)c1 C(C(=O)N1CC2CC2(C(N2CCN(C)CC2)=O)C1)(C(C)C)NC(CC(C)C)=O CC(C)C(CO)C(=O)NCC1CCN(C(=O)Cn2cc(Br)c(=N)[nH]2)C1 C=C(C)CC(C(=O)N1CCCN(C(N)=O)CC1)NC(=O)C(C)c1ccco1 c1(NCc2cn(C(C)C)nn2)cc(S(=O)(=O)N(CCCO)C(C)C)ccc1C#N CN1CCN(C(c2cnc3ccc(C#N)cn23)=O)c2ccc(Cl)cc21 Cc1cc(F)ccc1C(=O)NCC1COCC1NC(=O)CCSC1CCCC1 N1(C(C2CC(C)N(C)CC2)=O)CCN(C(C2(C(F)(F)F)CC2)=O)CC12CCC2 C(=O)(CC(C)SC)NC(CNC(CCC)=O)CC N1(C(c2ccc(CC)cn2)=O)CC2CC(C(N3CC(N4CCC4)C3)=O)(C2)C1 C1(CC)(NC(=O)C(C)S(C)(=O)=O)CCCN(C(c2cn(C)nn2)=O)C1 C(=O)(C1=C(C#N)CCC1)NCC(CN(C(c1cc2sccc2cn1)=O)CC)(C)C c1(N2CCC(NC(=O)CCc3ccncc3)C2)cccc(F)c1[N+](=O)[O-] S(=O)(=O)(c1cccnc1N1CC(O)CC(C)(C)C1)N(C)CC1CCN(CC)C1 C1(C(N2CC(CC(=O)NC(C#C)CCC)(OC)C2)=O)OCCCC1(C)C C1(C2CCN(C(=O)CC3CCCS3(=O)=O)C2)(NC(c2c(C)ccc(Cl)c2)=O)CC1 C1(C(N2CCC(O)(CN(C(c3cc(C)ncc3)=O)C)C2)=O)Cc2nncn2C1 N1(C(C2(C)CC2Br)=O)CC(C2CCN(C(c3coc(Cl)n3)=O)CC2)C1 N1(C(C2CCC(C)O2)=O)CCC(CO)(CNC(c2[nH]nnc2C(F)F)=O)CC1 N1(C(C(C)OCCOC)=O)CCCN(C(C2(C#N)CC(F)(F)C2)=O)CC1 C1(C(C)C)C(C(=O)N(C)Cc2nccs2)CCN1C(c1ccc(F)s1)=O c1(OCC(=C)C)ccccc1COC(C1CC(O)(CC(C)C)C1)=O.C=O N(C1CCCCc2cnn(C)c21)C(N1CCN(C)C(c2cccs2)C1)=O c1(OC)cnc(C(=O)NC2CCCC2NC(C2CC(O)C2)=O)c(F)c1 c1(C(=O)NCCCCNC(C(CC)OCC)=O)cc(OC)ccc1C(C)C C(=O)(C(CNC(=O)CC1(C)OCCO1)C(C)C)N(CC(C(=O)OC)C)C N1(C(=O)CCC2CCCOC2)CCC(O)(CNC(C2(O)CCOC2)=O)CC1 CN=c1[nH]c(=NCC2CCCC(O)C2)[nH]c(=NCc2cnn(C(C)C)c2)[nH]1 CC1CN(C(=O)C(C)CO)CC1CC(=O)NCc1nc(N(C)C)no1 CC1CC2CCCCC2N1C(=O)Cn1cc(-c2ccc3[nH]ccc3c2)nn1 Cc1ccccc1-c1ccc(C2(NC(=O)NC3CCC(=O)NC3)CCC2)cc1 N1(C(CCCCN(C)C)=O)CCC2(CCCC2NC(C2CCN(C)CC2)=O)CC1 C1(NC(c2c(CC)nccn2)=O)(CNC(c2ncccc2Cl)=O)CC2CCC1C2 C(=O)(CC(C)C(=O)NCCC(=O)N(C)C)OCC.C12CCCC(C1)C(=O)N2 c1(OC)nn(C)cc1C(N1CC=CC1C(=O)NCc1c(C)cnn1C)=O c1(C(N2C(CC(C)C)CC2)=O)coc(CNC(C2CCC(O)C2)=O)n1 C1(NC(C2CCS2(=O)=O)=O)C2CC3CN(C(c4ccnc5ncnn45)=O)C1C3C2 N1(C(c2c(C)cc(SC)s2)=O)CC(F)(F)CC1(C)CNC(=O)CCn1cccn1 C(=O)(CC(C(F)F)NC(=O)C1=CCOCC1)NC(CCC)CC CC1CC(C(=O)NCC2COCCN(C(=O)CC=C(Cl)Cl)C2)=NO1 c1(C(=O)NC2C(NC(c3cc(C)oc3C)=O)CC2)cnc(C(C)(C)C)nc1C CC1(C)CCC(C(=O)NC2(C)CCSC2)(NC(C2CCC(C3CC3)C2)=O)C1 N1(CCNC(C2CC(NC(C=CC)=O)C2)=O)CCCCC1=O C12(CNC(c3ccnn3CCF)=O)CN(C(=O)C=Cc3cnc[nH]3)CC1CCO2 C(=O)(C1CCCc2c(O)cccc21)N1CC(CNC(C(C)OCCOC)=O)C1 c1(NC(C2CCN(C(C(CC)CCOC)=O)C2)C)cc2nnc(C(C)C)n2cn1 CC1CCC(CO)CN1C(c1ccccc1)C(=O)NC1CCCC1 c1(NC(C)=O)ccc(C(=O)N(CCNC(C2CCC(C)S2)=O)C2CC2)c(O)c1 c1(C(=O)NCC23OC(C)C(C2)C3)ccnc2c1ccn2C NC1C2CCC3C(C2)C13C(N1CCN(Cc2cc3cnccc3[nH]2)CC1)=O Cc1c(Cl)nc[nH]c1=NCC1CC(CNC(=O)CC2(C)CC2(F)Cl)C1 C(=O)(CC(C)(C)C#N)NCc1ncc(C(=O)NCC(=O)N(CC)CC)cn1 N1(C(c2c(=N)[nH]cnc2)=O)CC2CC(C(=O)NCC3(CCO)CC3)CC2C1 c1(NC(CSCCCOC)=O)ccc(O)cn1 C12(C(=O)OC)CC(NC(=S)NCC3CCCC3N(C)C)(C1)C2 CC1CCC2(NC(=O)N(C3CN(c4ccncc4)C3)C2=O)c2ccccc21 c1(CCNC(=O)OC)ccc(S(=O)(=O)NCc2ccc(OC)cc2)s1 CC(CC(F)(F)F)N=c1[nH]c2c(c(=NCC3(CC(N)=O)CC3)[nH]1)COCC2 C1(CC(=O)NCC(C)NC(C2CCC(SCC)CC2)=O)CCCC2(CCC2)O1 C1(N(C(CCC#CC)=O)C)CN(C(c2cc3sccc3s2)=O)CCC1C c1(C(N2CCN(C(C(C)C3CCC3)=O)CC2)=O)nc(C(F)(F)F)n2ccncc12 N1(CCC(=O)NC2C(NC(C(C)(C)c3ncco3)=O)C2)Cc2ccccc2C1=O CCCC(O)C(=O)N1CCC1(C)CC(N1CCN(CC2CC2)CC1)=O Cc1cc(=NCc2ccc(C(N)=O)nc2)[nH]c(N(CC(C2CCCCC2)C)C)n1 c1(C(N(CCCNC(CNS(NC)(=O)=O)=O)C)=O)cc2c(C)ccc(F)c2o1 c1(SCC(=O)NC2CCN(CC(N3C(C)CCCC3)=O)C2)nnc2ccccn12 C1(C(CNC(CC)=O)(C)C)CCCCN1C(c1cc(Br)oc1C)=O C1(C)(C(N2CC(C(C)NC(c3ccc(C)o3)=O)OCC2)=O)CCCNS1(=O)=O c1(NC(c2c(CC)cccc2)C(=O)Nc2ccccc2CO)ccc(C)c(F)c1 c1(NCC(C)C(C)(C)C)cc(S(=O)(=O)NCC2COC(C)(C)CO2)ccc1C#N C(c1cccc(F)c1)=CC(=O)N(CCCNC(CCCc1nnc(C)n1C)=O)C C(=O)(C1=C(Cl)CCC1)N1C(CC)C(C(=O)Nc2cn(C)nc2C)CC1 N1(C(CNc2n(C)ccn2)=O)CCN(C(C2CC2CF)=O)C(c2ccccn2)C1 c1(C(N2CCCC(N(C(CN3CC(C)C3)=O)C)CC2)=O)ccc2ccnn2c1 c1(C(=O)NC(C(C)C)(C)CNC(c2ccnc(O)c2)=O)ncn2c1CCCC2 C(CCN(C(=O)C(F)(F)C12CC(C1)C2)C)(C(C)C)NC(c1c(C)ncs1)=O C1(C(N2CCCCC(NC(C(C)OC)=O)C2)=O)CSC(c2ccccc2)=N1 C(=O)(C1CCCc2c1ncn2C)N1CCCC(CNC(C(C)OC2COC2)=O)C1 C1(C)(CNC(C(C)N(C(=O)C(C)OC(C)C)CC)=O)CCCC1O c1(C(=O)NCCCC(C)(C)NC(C2CC2C2CC2)=O)ccc2ncnn2c1 CCCC(C(O)C(=O)NC1(C)CCCOC1)NC(=O)CN(CC(C)(C)C)C C1(NC(=O)CO)CS(=O)(=O)CC1NC(=O)Cc1cscc1Br C1(CCNC(C(C)N(C(C2CCC3(CCC3)C2)=O)C2CC2)=O)OCCCC1(C)C c1(C(N(CCNC(c2cc(OC)ncc2)=O)C2CC2)=O)c(C)ccc(Cl)c1F C1(CC)C(O)CCN1C(c1cccc(F)c1)C(=O)NCCC1(C)CC1 N1(C(CC(=O)OC)=O)CCC(NC(c2ccc(CC(F)(F)F)cc2)=O)CC1 Cc1ccc(C)c(C(=O)NCC2C(C)CCN2C(c2cccc(C)c2Cl)=O)c1 c1(CC)ccc(NC(=O)CCOc2ccccc2OCC(=O)NC)c(C)n1 N1(C(c2c(C)ccnc2)=O)C2CCC(C2)C1C(N1CCCC1c1ncc[nH]1)=O c1(CC)n[nH]cc1C(=O)NC1CCCC1NC(C12CCCC1C2)=O c1(CN2CC(C(=O)Nc3c(C)ccc(Br)n3)SCC2)nc2ccccc2s1 c1(CC#N)cccc(C(N2CC(O)CC2C(=O)NCC2CCC(=O)O2)=O)c1 C1(CNC(C2CC(NC(C(=Cc3ccco3)C)=O)C2)=O)CC(O)C(O)C1 c1(OCCC)cccc(CNCC2(CC(=O)NC(C)=O)CCC2)c1F C1(C2CCCN(C(c3cc(F)cc4ccoc34)=O)C2)(NC(CC(C)OC)=O)CC1 C1(NC(c2cncc(C)c2)=O)CCCC(N=c2nc(Cl)[nH]c(C)c2C#N)C1 C1(CNC(c2n(CC=C)ccn2)=O)CC2(CO1)CN(C(C1CCSCC1)=O)C2 CC(C)(C)CC(O)C(=O)NC1CC=C(C(=O)N2CCCCC2)C1 c1(N(CCNC(C(c2ccccc2Cl)OC)=O)C(C)C)ncc2c(n1)CCCCC2 N1(C(C2(C(C)C)CC2)=O)CC(O)(C2CCN(C(=O)C(c3cccnc3)O)CC2)C1 N1(C(CC2N(C(c3cc(CC)ncc3)=O)CCCC2)=O)CCC(OC)C(C)(C)C1 C1(NC(C(C(C)C)NC(C2ON=C(CC)C2)=O)=O)CCCCCC1O C1(CNC(C2(C(C)C)CC2)=O)CCC2(CN(C(=O)CCOCC3CC3)C2)O1 Cc1ccc(Cl)c(C(=O)N(C)CC2CCCCN2C(c2cnncc2C)=O)c1 C1(NC(CC2(N(C(c3c(C)cn(C)c3)=O)C)CC2)=O)CCOC2(CCC2)C1 C(=O)(C#CC1CC1)NCC(C)(C1CC1)NC(=O)CCN1CCN(S(C)(=O)=O)CC1 c1(N2CCCC(O)(CCO)C2)ncnc2c1ncn2C1CC1C(F)(F)F C1(C(=O)NCC(CN(C(C(C2CC(C)(C)C2)OC)=O)C)(C)C)CCCS1(=O)=O C(=O)(C(O)P(C)(C)=O)N(CC(C)(CN(C)C)NC(C)=O)C1CC1 C12(CNC(CC(=O)N(C)C)=O)CC3CC(CC(NC(C4CCNC4=O)=O)(C3)C1)C2 C1(N(C)C(C2CC(C(F)(F)F)C2)=O)CCCCN(C(c2cncc(F)c2)=O)C1 CCCC(CCC)C(=O)NC1C=CCN(C(C2CC2c2cccc(O)c2)=O)C1 C(CC(C)CCNC(c1cc(OC)ncn1)=O)NC(C1(CCC)CCC1)=O Cc1nnc2c(C(N3CCCC(NC(c4cncn4C)=O)C(F)C3)=O)cccn12 N1(CC(=O)NCC2CN(C(C3CCC(C(=O)OC)C3)=O)C2)CCCCCC1=O c1(OCC(=O)NCC(CC)Nc2cc(C)nc(C3CC3)n2)cccc(C)c1F N1(C(C(C(C)C)C2CCC2)=O)CCC(C(=O)NOCC2(C)CCC2)CC1C CC1CC(c2cn(CCNC(N)=O)nn2)CCN1C(=O)C(F)C1CCCC1 c12ccc(c(OC)c1)c(=O)[nH]2.N1(CC)CCN(C(=O)Cc2nncn2C)CC1 c1(OCC)ccc(Cl)c(C(N2CCC(N(C(=O)COCC)CC3CC3)CC2)=O)n1 O=C1CC(C(N2CCC(C(F)C(=O)NC3CCCCC3(F)F)CC2)=O)NC(=O)N1 C1(NCc2ccccc2)CC(=O)N(C)C1.C1(c2cc[nH]n2)C(=O)NCC(C)N1C C1(C(C)(C)C)CN(C(=O)Nc2ccc(F)cc2)CCN1Cc1ncsc1Br N(C(=NCc1nccc(C(F)(F)F)n1)NCC1(C)COCCO1)CC(C)(C)C c1(CNCC2CCCC(C(=O)OC)C2)cc2n(n1)CCN(C)C2 CCCC(CCC)CC(=O)NCC12CCC(CN(C(C3(C)CNC(=O)C3)=O)C1)C2 CC(C(C)(C)NC(c1cc(F)c[nH]1)=O)NC(c1cncn1C)=O C(=O)(N=c1[nH]nc2[nH]ccnc1-2)c1c(C)nc(NC(CCC#C)=O)s1 Cc1ccc(C(=O)N(C2CCN(CCCN3CCCC3=O)CC2)C)cc1Cl C1(CN(C(=O)CCOCC2CC2)C)CCCCN1C(=O)CC1CCC1(F)F C1(SC)CN(C(C2CCCC(C3CC3)O2)=O)CC1NC(=O)CC1SC(=N)NC1=O C1(CCC=C)CCCN(C(=O)C(C(C)C)N(C(=O)COCCF)CC)C1 c1(C(C(=O)NC2CCC2)N(c2ccc(C)cc2)C)cccc(SC)c1 CCCC(CC(C)C)C(=O)NC1CN(Cc2ccsc2)CC1(C)C c1(C(N(CCNC(C(C)CC(C)(F)F)=O)C)=O)nc[nH]c2ncc(Br)c1-2 N1(C(C2OCCN(CC)C2)=O)CCC2OCCN(C(=O)Cn3cc(C)cn3)C2C1 N1(C(C(CC#C)O)=O)CC(NC(C2(CCCC)CCC2)=O)CC12CCOCC2 c1(OCCCC)ccc(C(=O)NCC(C)NC(C2C(C)C2(F)F)=O)cc1 Cc1ccc(F)cc1CC(=O)NC1CCC(NC(c2n[nH]cc2[N+](=O)[O-])=O)C1 Cc1cc(C(=O)N(CCC(C(C)C)NC(=O)C(C)N2CCC2)C)cc(O)n1 c1(C(N2CC(NC(Cc3cn(C)nn3)=O)C(F)C2)=O)cnc2ccccc2c1 N1(C(C2N(S(C)(=O)=O)CCC2)=O)CC2C(NC(C34CC(CC5CC5)(C3)C4)=O)C2C1 C1(CC(N2CC(OC)(CNC(=O)C(O)CN(C)C)C2)=O)Cc2cc(Cl)ccc2O1 c1(C(=O)NC2COCCN(C(C=CC=CC)=O)C2)cc(O)nc2c1CCCC2 C1(C(=O)NCCC2N(C(CC(C)N(C)C)=O)CCSC2)CCc2nncn2C1 C1(NC(CCCN=[N+]=[N-])=O)CCCCC12CCN(C(c1ccc(F)nc1)=O)C2 C(CCCCCS(N)(=O)=O)NC(C(C(F)(F)F)NC(C(C)C)=O)=O Nc1ccc(C2=CCN(C(=O)N=c3nc(C(F)F)s[nH]3)CC2)s1 C=Cc1ccc(C(=O)OC2CCCN(c3nc(C)ncc3F)C2)cc1 C1(C(=O)NCCN(CCO)CC)CCC(C)(C)N(C(=O)C(c2ccn(C)c2)C)C1 N1(C(=O)CCc2ccccc2O)CC2(CCN(C(C3(F)CCCOC3)=O)C2)C1 C1(NC(Cc2nc(C)[nH]n2)=O)COC2C(NC(=O)CS(N)(=O)=O)COC12 CCC(C)C(O)C(=O)N(C)CCN(C(=O)C(=O)Nc1ccc(F)c(C)c1)C C1(NC(c2c(C)cc(SC)o2)=O)C(C)CN(C(c2cc(C)sn2)=O)CC1C N1(C(C(F)=CC)=O)CCN(C(=O)Cc2cc(C)sc2C)CC1c1cccnc1 C1(NC(C2CC(SC)C2)=O)CC(C)CN(C(c2cc3occc3[nH]2)=O)C1 C1(C(F)(F)F)(NC(C2CCN(C(=O)CN3CCOCC3)CC2)=O)CCCCC1 C1(NC(C2C(OCC)CC2)=O)CC2CCC1(C(=O)NC1CCCSC1)C2 C1(C(N(CCCCN(C)C)C)=O)C2CC3C(C2NC(C2CCCC(CF)C2)=O)C13 N1(C(C(CC)N(CC)CC)=O)CCC2CC1CN(C(C1C3(CC3)C13CC3)=O)C2 c1(NC(CN(C(C(C)OCC#C)=O)CC2CC2)=O)ccc(O)c(F)c1 Cc1ccc(C(N2CCCC(NC(C3CN(C4CCC4)C3)=O)C2)=O)cc1C CC(C(C)(C)NCC(N1CCCCC1)C)c1ccccc1 C1(C(=O)NOCC)c2ccc(cc2)N1.C(CC1CC1)OCC C1(F)(C(N2CCC(N(CCC)C(C3(C(F)(F)F)CCCC3)=O)C2)=O)CCOCC1 C1(NC(=O)C=CSCc2ccco2)CC12CC(NC(=O)C(F)C1CCC1)C2 CCC(CC)C(F)C(=O)N1CC(O)(CNC(=O)CC(C)C(=O)OC)C1 C(C(CC(C)(C)C)N=c1c(F)c[nH]cc1F)OC C1(C(N(C2(CN(C3CCOC3)C(c3[nH]cc(C)n3)=O)CC2)C)=O)CC(F)(F)CS1 c1(C(=O)NC2C(CNC(CN(CCC#C)C)=O)C2)c(C)nsc1NC1CC1 C1(NC(=O)C(C)(O)C2CC2)CCN(CCC(C)C)CC1.C1(C)C(=O)N1 C1(NC(C2C(C)(C)CC2)=O)CC2CC(NC(=O)CCc3cncc(F)c3)C1C2 CCCC(C)(C)CC(=O)N(CC(CC)NC(c1ncc(F)cc1N)=O)C N1(C(C(c2cccs2)SC)=O)CC(NC(=O)CC2(n3cccn3)CC2)C(C)C1 C1(N(C(c2cnc(O)s2)=O)C(C)C)CC(Nc2ncccn2)CC1O N1(C(CC(CC(C)C)C)=O)CCCC2(C1)CN(C(c1cccc(C#N)c1)=O)C2 N(C1CCc2ccc(Cl)cc21)C(C1CCCN(C2CCN(CC)C2=O)CC1)=O c1(N(CCOCCC)C)nc(C)cc(=NCC(=O)Nc2cc(C)oc2C)[nH]1 C1(OC(c2cn(CC(F)F)cn2)=O)C=CCCC1C=O.CC(C(=O)O)=C1CC1 S(=O)(=O)(c1cc(C(N2CCN(C(=O)CCC(F)F)C(C)C2)=O)n(C)c1)NC N1(C(c2c(C)snn2)=O)CCC2(NC(=O)CN3C(=O)CCCC3=O)CC2C1 N1(C(C)=O)CCCCC1C(=O)NC1CN(C(=O)OC(C)(C)C)CC1O C(=O)(C1c2c[nH]nc2CN1C(c1ccc(C#N)s1)=O)NCC=CCCOC CCC(CC(=O)NC(c1ccccc1)C(=O)NCC(C)(O)CCO)C1CCC1 CC(C)CC(=O)NCC(C1CCCC1)NC(=O)Cn1cc(C(C)O)nn1 C(=O)(C(F)(F)C=C)N(CCCNC(C1(CC#C)CCOC1)=O)CC C1(CNC(CCOC(C)=O)=O)CCN(C(C2CC(F)(c3ccccc3)C2)=O)C1 C1(CNC(c2[nH]cc(CC)c2)=O)CN(C(=O)Cc2cc[nH]n2)CC12CCC2 c1(CC)cc(C(=O)OC)ccc1NC1(c2cccc(C(F)(F)F)c2)CC1 N1(C(C2(COC)CC2)=O)CCC2(CCCN(C(=O)CC(C)(O)COC)C2)C1 C12(C(=O)NCC3(OCC)CCC3)CCCC1CC2 C=C(C)CN=C(NCc1cc2ccccc2[nH]1)NCC1CCN(CC)C1 C1(C(=O)NC(c2ccsc2)C)CN(c2ncc(-c3ccccc3)cn2)CCC1O N1(C(C(CC)C)=O)CC2OCCN(C(=O)Cc3cccc(Cl)c3F)C2C1 c1(CNC(C(C)NC(c2cccnc2)C(=O)OCC)=O)nnc2ccccn12 c1(C(N2CCC(CNC(c3ccc(CC)[nH]3)=O)C(C)C2)=O)cc(C)c(Cl)cc1C CCC(C(=O)N(CC(C)N(C)C(C1CC(c2ccccc2)C1)=O)C)C(C)(C)CC N1(C(c2cccc(O)n2)=O)C2CCC1C(C(N1CC3CC3C1)=O)C2 C(CCCC(=O)NCc1cccc(NC(=O)CN2CCOCC2)c1)N(C)C c1(C(=O)NC(COCC)C(=O)NC2CC=CCC2)cnccc1C#N Cc1nn(C)cc1C(C)C(=O)NC1CC1NC(c1ccncc1C(F)F)=O C12(CNC(C3CC3(F)F)=O)CCC(CN1C(c1cccc(-c3nccs3)c1)=O)C2 N1(C(CC(C)OC)=O)CCC(C(C)(C)NC(=O)C(C)Cc2cnn(C)c2)CC1 c1(C(N2C(C(=O)Nc3cc(C)nc(Cl)c3)CC3(CC3)C2)=O)cn2cc(Cl)ccc2n1 C1(COC)CN(C(=O)CCC2CC2(Cl)Cl)CCN1C(=O)C(c1cccn1C)=O C(=O)(CCCc1nc(C)no1)N(CC(CC)NC(=O)Cn1nnc(=O)[nH]1)C c1(C(=O)NCC(C)N(C)C(C2(C)CCCS2)=O)ccc2[nH]c(=N)n(C)c2c1 CC1=C(C(=O)NCC2CCN(C(c3nccc(Cl)c3O)=O)C2)CCC(C)(C)C1 N1(C(C(C)c2cccs2)=O)CCN(C(=O)CCC2CCC(=O)NC2)CC2(CC2)C1 c1(OC(C)C)ccc(NC(C2CCN(C(c3ccc(C(=O)O)s3)=O)CC2)=O)cn1 c1(C(N(C2CCC(NC(Cc3c(C)noc3)=O)C2)C)=O)cnc2[nH]cnc2c1 CCC(O)C(C)C(=O)N(C1CCN(C(c2cnc(OC)nc2C)=O)CC1)CC C1(C(=O)NCC(CNC(C2(OC)CCSC2)=O)(C)OC)CC(C(C)C)=NO1 C(C(CO)C(F)(F)F)NC(C(c1cnn(C)c1)NC(c1cn(CCC)nn1)=O)=O N1(C(CCOCC#C)=O)CC2CCC1C2NC(=O)CCS(C)(=O)=O N1(C(C(CCOC)C)=O)CCC2(CCCN2C(=O)Cn2ccc(C(F)F)n2)CC1 c1(C(=O)NCCC(CNC(c2cc(CC)ncc2)=O)O)nc(C)ncc1Cl c1(C(N(CC(CC)NC(c2sccc2CO)=O)C)=O)cc(CO)on1 c1(OC)cnccc1C(N1CC(CNC(C2COC(C)C2)=O)(OC)C1)=O CCC(CCOC)C(=O)NCC(C)N(C(=O)CC1SC(=N)NC1=O)C C(CCCC(=O)NC1(C(N2CC3C(C)C3C2)=O)CCN(C)C1)SC c1(SC(C)C(=O)NCCNC(c2c[nH]nc2-c2ccncc2)=O)ccccc1Cl C(=O)(C(CNC(c1ccc(F)cc1F)=O)C(C)(C)C)N(C(CC(=O)OC)C)C C=CCC(C)(CC)C(=O)NC1CC(C)CN(C(c2cccc3nncn23)=O)C1 C(CSc1ccc(Cl)c(Cl)c1)(C(C)(C)C(C)C)OCC Cc1nc2c(s1)CCCC2C(=O)NC(C)CNC(c1cncc(F)c1Cl)=O N1(C(c2c(SC)cccc2)=O)CC(NC(c2cc(C)ccc2F)=O)CC2(CC2)C1 N1(C(C(CC)OC)=O)C2CCC1C(C)C(NC(c1ccc[nH]1)=O)C2 c1(C(N2C(C)C(NC(=O)CCc3cccc(O)c3)CC2)=O)ccc(F)c(Cl)c1 C1(NC(C2(OC)CCOC2)=O)C2CC1N(C(c1cc(C3CC3)nn1C)=O)C2C c1(NC(COC)CCO)[nH]c(=NCc2cc(Cl)ccc2OC)nc2c1cnn2C C1(NC(C2C(C)C2)=O)CC2CCC(C1C)N2C(C1CC2CCCCN2C1)=O c1(C(=O)OC)cc(C(=O)NC2CC(C)N(C(=O)C(c3cnn(C)c3)C)C2)ccn1 C1(C(N(C2CCN(S(C)(=O)=O)C2)CC(C)C)=O)CCN(Cc2ccccc2Cl)CC1 N1(C(C(C)OCC)=O)CCCCC2(CCN(C(C3(C4CCC4)CCC3)=O)C2)C1 CC1=C(C)CC(C)(C(=O)NCC(C(C)C)NC(C2(C)CCCC2)=O)CC1 N1(C(CCCN(C)C)=O)CCCC(CNC(=O)CCCN2CCCC2)CC1 C(CCCCC(=O)NC(CCN(C(=O)CC1CCCOC1)C)C(C)C)OC c1(SCCC(=O)NC2(CCNC(=O)C(F)C3CCC3)CCC2)ccccc1 C1(C(=O)NCC2(CC)CC2)CCC2(CN(C(c3cc(-c4ccccn4)[nH]n3)=O)C2)O1 N1(C(c2cc(SC)oc2)=O)CC(CNC(=O)C(C)(C)C(C)C)C2CCCCC12 c1(C(=O)NCCN(C(=O)CN2CCC2C)C(C)C)ncc(Cl)cc1Cl N1(C(C=Cc2ncc(C)[nH]2)=O)CCCCC1C1CCCN1C(c1ccc(C)s1)=O C(=O)(C#CC1(C)CCCO1)N(C(C(=O)NCC1ON=C(CC)C1)C1CC1)C C1(C(NNC(=O)NCCCC#C)=O)C2Cc3cc(Cl)ccc3C12 N1(C(=O)NCC2(C(F)(F)F)CCC(OC)C2)CCC2(C=CCO2)C1 C(=O)(CCC(F)(F)F)NCC1CN(C(c2ccc(CC)[nH]2)=O)CC1C Cc1csc(CC(=O)NC2CC(F)(CNC(=O)C(C)CC3CCC3)C2)c1 N1(C(C(C)(C)O)=O)CCC2(CCCN2C(c2cccc3c2OCC3)=O)CC1 CCCCCCCC(=O)NCC1(NC(c2sccc2OC)=O)CCC(C)(C)CC1 C1(C(=O)NCCN(C)CC)(CO)CCN(C(=O)CSCCC(C)C)C1 c1(C(N(CCCCCNC(C(C=CCCC)O)=O)C)=O)ccc(CO)nc1 CC1CCCCC1OCCNC(=O)CC(C)(C)n1cc(C(C)(C)C(N)=O)nn1 C1(C(C2(C(=O)NCC(C(C)C)NC(=O)OC(C)(C)C)CC2)=O)CCCCC1(F)F C(N=c1[nH]c(=NCc2cncs2)c2ncccc2[nH]1)c1ccc(SC)nc1 c1(C(N2C(C(=O)Nc3ccc(C)cc3)CC(C)C2)=O)cc(Br)nc(Br)c1 C#CC1(C(=O)NC(C)CC(C)O)CN(C(=O)CCc2ccco2)C1 N1(C(c2c(OC)cc(C)s2)=O)CCC2(C1)CN(C(C13CC(C)(C1)C3)=O)C2 CC#CCC(C(=O)NC1CCC(O)CC1)NC(c1cn2c(n1)CCC2)=O N1(C(c2c(C)scc2)=O)CC2(C1)CN(C(C1(C3CCCCO3)CC1)=O)CCO2 c1(C(N2CCOCC(NC(C(CC)C)=O)C2)=O)cc(C#N)c(O)nc1N C12(CC(=O)NCc3cccc(NC(c4occ(C)c4)=O)c3)CCC(CC1)OC2 Cn1ncc(C(N2CCC(C3CCCN3C(=O)CO)CC2)=O)c1F c1(SCC)ccccc1C(=O)NCCCCN(C(=O)CCC(=O)N(C)C(C)C)C C1(CNC(C(=O)NCCOC)=O)CC(C)(C)CN1C(c1cncc(F)n1)=O Cc1onc(C(F)(F)F)c1C(N1CCN(C(C2CCN2C2CCCC2)=O)CC1)=O N1(C(C=CC(C)=O)=O)CC(C2CCCCN(C(c3nncn3C3CC3)=O)C2)C1 C(C(O)CC(=O)N1CCCC(CN(C)C(c2cc(C(N)=O)cs2)=O)C1)N(C)C c1(C(=O)N(C2CC2)Cc2noc(C3CC3c3ccccc3)n2)ccc(Cl)cn1 CCC(C(=O)N1CCC(NC(C2(C)COC(=O)OC2)=O)C1C)C(C)C C1(N(C(=O)CCCc2ncco2)C)CN(C(c2cc(O)ncn2)=O)CC1F c1(C(=O)NCC2C=CCN2C(=O)CC2CCCC2O)cncc(Cl)c1 c1(C(N2CCOCC(CNC(CCOCC)=O)C2)=O)cc2ccc(OC)cc2[nH]1 C(=O)(CCC(F)(F)F)NCCN1CCC(NC(C(N2CCCC(O)C2)C)=O)CC1 N1(CC(C)NC(=O)CC(C)(C)C)CCN(C(=O)CC(C)N(C)C)CC1 c1(CCC(=O)NCC2(CCNC(C(CC)F)=O)CC2)ccc(C)cc1C c1(OC)ccc(Cl)cc1C(N1CCC(NC(=O)CC2CC2(Cl)Cl)C(F)C1)=O N1(C(C2C(C)C2)=O)CCOC(CC(N2CC(CC3CCCC3)C2)=O)C1 C1(NC(CN2C(=N)NCC2)=O)CCCC2CN(C(C3(F)CC=CC3)=O)CC12 CCC(C)(C(=O)N1CC(CNC(c2ccncn2)=O)C(C(F)(F)F)C1)C(N)=O CCC(CC(F)F)C(=O)N1CCOCC1CNC(c1nn(CC)cc1Cl)=O N1(C(C2CCCC2)=O)CCC(O)(CCO)CC1.C1(CC=C)(C(=O)N)CC1 CC(C)CC(CNC(c1cccnc1S)=O)C(=O)N1CC(c2ccncc2)C1 C1(CC(=O)NC2(C(=O)NC(C3(OC)CCC3)C)CCC2)COC(=O)C1 N1(C(C2OCC(C)C2)=O)CC2(CCCC2NC(c2cccc(CN(C)C)c2)=O)C1 CC1(NC(C2CC=CCC2)=O)CN(C(c2ccsc2)=O)C1 c1(C(=O)NCCCCN(C(=O)CC(C)(C)O)C)cc2cc[nH]c2cn1 C1(C(N2CCOC(C)C2)=O)(OC)CCN(Cc2ncon2)CC1 c1(C(=O)NC2CN(C(C3N(C(C)=O)CCCC3)=O)C2)ccc(N)c(C)c1F c1(CC(C(=O)NC2C(CNC(C=CCOC)=O)COC2)F)ccc([N+](=O)[O-])cc1 c1(C(=O)NC2(C)CCCC2)ccc(NCCNC(=O)CP(C)(C)=O)cn1 CC1CC2CN(C(C3COCCC3NC(C3CCC(CO)CC3)=O)=O)CC12 C1(CNC(C2(SC)CC2)=O)CN(C(c2coc(CO)c2)=O)CC1C(F)(F)F c1(C(=O)NC2CC(NC(C3CCC(NC(CC)=O)C3)=O)C2)ncccc1S(C)(=O)=O CCCC(CCNC(C1CC(NC(=O)Cc2csnn2)CCO1)=O)CCC C12(C(N(CC(COCC)O)C)=O)CC(CN1C(C1CC=CCC1C)=O)C2 N1(C(CC=C)=O)CC(NC(=O)C(C)N2CCC2)CC1(CC)CC C(=O)(C1=CCCOCC1)NC1CCCC(CNC(=O)Cc2ccns2)C1 Cc1ccc(C(=O)NCCCC(C)NC(C2CC2c2cccnc2)=O)nc1 C1(N(C(C(c2cncc(Cl)c2)OC)=O)C)CC(NCCSC)C12CCC2 c1(NCc2cc(OC)ncc2)nc2ccccc2nc1NCC(C)OC(C)(C)C N1(C(C)=O)CCCN(C(C2CC3(Cc4ccc(Cl)cc4)CCCC23)=O)CC1C c1(COC)nc(=N)[nH]cc1C(=O)N(CC(CO)(CO)NC(C1CC1C1CCC1)=O)C C1(N(C)C(c2cn(C3CCCC3)nn2)=O)CCCC(N(C)C(c2csnn2)=O)C1 CCCCCCCCC(C)C(=O)N1CCCC(C2(NC(=O)CCC(F)F)CC2)C1 c1(C(N(C2CC(NC(C3OCCC3(C)C)=O)C2)C)=O)ccc(O)cn1 S(=O)(=O)(c1cnn(C2CC2)c1)N(C)CCc1cccnn1 c1(C(=O)NCc2occ(C(=O)NCC(C)(O)C(F)F)n2)cccc2cc[nH]c12 c1(C(C(=O)NCC(C)C)N(CC(=O)NC)CC=C)ccc(C(F)(F)F)cc1 C1(CNC(CC(C)F)=O)CC2CCCC2N1C(=O)C(n1cc(Br)cn1)C C1(NC(CC2(OCC)CC2)=O)CCCC1NC(c1sccc1COC)=O C1(CNC(=O)COc2ccsn2)CCN(C(=O)CC2CCCS2(=O)=O)CC1(F)F C1(CNC(C2(C#C)CCCC2)=O)CC(C)CN(C(c2[nH]ccc2CC)=O)C1 N1(C(C(c2cccc(O)c2)C)=O)CCC(NC(c2cccc(O)n2)=O)C1(C)C N1(C(c2c(C)nc(CCC)o2)=O)CCC(NC(C2CC2C(C)C)=O)C2(CCC2)C1 C(C(O)C(F)(F)C(F)(F)F)Nc1nccc(=NCC2(C)CCOC3(CCC3)C2)[nH]1 C1(NC(c2ccccc2)=O)(CNC(c2cnc(C3CC3)s2)=O)CC2CCC1CC2 C12(NC(CCn3c(C)csc3=O)=O)CCC(CC1)N(C(=O)C(O)P(C)(C)=O)C2 C1(CC(=O)NCC2N(C(Cc3c(C)cco3)=O)CCCC2)CCCCCC1(F)F C(=O)(CC1=CCN(C)CC1)N1CC(NC(c2ncc(Cl)cc2Cl)=O)CC(C)C1 C(=O)(CC1C(=O)Nc2ccccc21)NC1C(NC(C(C)OC(C)(C)C)=O)COC1 CC(CC(=O)NC1(C(N2CCC(C3CC3)CC2)=O)CC(O)C1)C(F)(F)F C(=O)(N=c1nc(Cl)nc2[nH][nH]cc1-2)C1(C)CCN(C(c2c(C)c(I)ccc2)=O)C1 CC1(C)CC(C)(C(=O)NC2C3CC(NC(c4ccon4)=O)CC23)C1 N1(C(C=C(CCC)CCC)=O)CCC(NC(=O)C(C)OCC2CC2)C(CO)CC1 C1(NC(C(n2cc(Cn3cccc3)nn2)C)=O)CCC2C1C2(F)F C(=O)(CCCC(C)CC)NC1(CC)CCN(C(=O)CCC(=O)c2cccs2)CC1 CC(C(=O)N1CCC(C(=O)NCCCN2CCCC2)O1)=CC1CCCC1 C1(CNC(CC2CCC(C)C2)=O)CN(C(c2c[nH]cc2C(C)(C)C)=O)CCCO1 C1(NC(C2(C#N)CCCC2)=O)CC2CCC1N(C(=O)CCN1CCNC(=O)C1)C2 N1(C(C(CC)n2cncn2)=O)CCC(CC)CC1C(=O)NCc1ccc(F)cn1 N1(C(C(C)NC(C)=O)=O)CCSCC1C(=O)NCCC(C)C N1(C(C(c2cc(F)ccc2Br)C)=O)CCn2c(C3CCC3)nnc2C1 C1(C(=O)NC(CCOC)CNC(=O)C=CSC)CCS(=O)(=O)C1 CCN=c1[nH]c(CNC2CCC(C(N3CC(O)C(F)C3)=O)OC2)cs1 C1(NC(CC)=O)CCC(NC(=O)C(=O)Nc2ccc(CC3CC3)cc2)CC1 C1(CNC(c2occc2C2CC2)=O)CC2CCC1N(C(=O)C(F)=C1CCC1)C2 N1(Cc2cn(C(C)CNC(c3ccc(Cl)cn3)=O)nn2)CC(O)CCC1=O N1(C(c2nc(C)sc2C)=O)CCC(C)(C)C1C(=O)NCCCC(=O)NC1CC1 c1(C(=O)NC2C(CNC(=O)C=CSc3ccccc3)COC2)cc([N+](=O)[O-])c[nH]1 c1(C(N2CCCCC2C2CCC2)C(=O)NCCC(=O)OCC)cnc(SC)n1C C1(CCC)(NC(C2CC2C)=O)CCN(C(=O)C(F)(F)c2cnn(C)c2)CC1 CC(C)(O)C(F)(F)C(=O)NC1CCCC1NC(c1cc(F)ccc1N)=O N1(C(c2ccccc2OCC)=O)CCOC2(C1)CN(C(c1cc(C#N)cs1)=O)C2 C=CCC(C)(C)C(=O)N1CCN(C(c2cc(-c3ccccc3)on2)=O)CC1CO n1(CC(N2CC3(CN(C(C4(OC)CS(=O)(=O)C4)=O)C3)C2)=O)ncc2cccnc12 c1(CC)ccccc1C(N1CC2C(C(=O)NC(CO)CCC3CC3)C2C1)=O C(C(C)CC(F)(F)F)NC(C1(c2ccc(C)nc2)CCC1)=O c1(C(C)NC(=O)NCCNC(c2cccc(Br)c2)=O)cccc(F)c1F c1(OC)cccc2c(CNC(c3cccc(Br)c3)CSC)cccc12 Cn1nc(C(=O)NC(C)(C)C=CC(=O)NCCN2CCCC(O)C2)cc1F N1(C(Cc2ccn(C)n2)=O)Cc2ccc(O)cc2CC1C(=O)NC1(C)CC1 c1(C(N2CCCC2c2nccs2)=O)cc(S(=O)(=O)Nc2ccc(Cl)c(Cl)c2)n[nH]1 N1(C(c2c(-n3cccn3)cccc2F)=O)CCN(C(=O)C2CC2)CC(CO)C1 N1(C(c2ccc(OC)nc2)=O)CC(NC(=O)Cc2cscn2)CCC(O)C1 CC1CN(C(C2C=CC(NCc3ccc(O)cc3Cl)C2)=O)CCN1C C1(CNC(C(F)=C(C)C)=O)CN(C(C2CCOCC2)=O)CC2(CCC2)O1 c1(C(=O)NCC2N(C(C3=CC(C)CC3)=O)CC2)c(Br)ccc(Cl)c1F c1(C(N(C(C=C)C)C)=O)cc(CNC(=O)C(C)C2CCCO2)cs1 C=CC(CCC)CC(=O)NC(C)CNC(c1c(C)cc[nH]c1=N)=O c1(C(=O)NC2C(NC(C(F)OC)=O)CCC2)cc(Cl)cn1C Cc1ncc(C(=O)NCC(C)CNC(=O)CC2CCC(C)C2)n1C N1(C(C2CC23CC(O)C3)=O)CCN(C(=O)Cn2cc(C(F)F)cn2)C(C(F)F)C1 c1(NC(CNC(=O)CCc2ccncc2)=O)cnc2ncnn2c1 C1(NC(C2C(C)CC2)=O)CCN(C(c2ccc(C#N)n2C)=O)C12CC2 c1(C(=O)NC2CN(C(C=C(C)c3ccco3)=O)CC2C)cc2cc(F)ccc2s1 CCC(CNC(=O)C(CN(C)C)NC(=O)CCOCCOC)(CC)CC CCC(C(=O)NCC1(C(=O)NCCc2cc(C)no2)CCCO1)SC c1(C(=O)NCC(CNC(C(CC)C#N)=O)O)cc2ccccc2oc1=O C1(CC)CCN(C(=O)Cc2scnc2C)C1C(=O)N(C)CCN(C)C(C)=O N1(C(CCOCC)=O)CCC2CCN(C(c3ccnc(CC)c3)=O)CC2C1 Cc1nc(C(N2CC(F)(C(=O)NCC3=CCCCC3)C2)=O)c(C)s1 c1(CC)ccc(C(N2CC3CC3C2CNC(C2CC(C)=NO2)=O)=O)nc1 c1(C(=O)NCC(C)NC(c2ccnc(OC(F)F)c2)=O)ccc(C(C)(C)C)cc1 CON(CCC(=O)NCC1CC12CCOCC2)C(=O)C(C)N(C)C C1(N(C(COCc2cc(C)no2)=O)C)CCCC(NC(=O)CCC2CCOC2)C1 Cc1ccc(Br)c(C(N2CCCC(NC(c3c[nH]cc3C)=O)C2)=O)c1 c1(C(=O)NC(C(C)(C)C)CNC(C2CC3(C2)CC3F)=O)ccc2c(c1)CCCO2 Cc1cc(C)c2cc(C(N3CCC(C4CCNC4)C3)=O)[nH]c2c1 c1(C(=O)NC2C(CNC(C(C)(C)c3cnsc3)=O)C2)ccc(C(N)=O)cc1 C12(C(=O)NC(CNC(C=C(CCC)C)=O)CCOC)CC1COC2(C)C CCCC(C)CC(=O)N1CCC(N(C(c2cc(C(=O)O)ns2)=O)CC)C1 c1(OC)ccc2c(c1)CCCC(Sc1nnc(C)n1CC(N)=O)C2 c1(C(=O)NCC2CCC(NC(CC=C(C)C)=O)CC2)cc(C)c2ccccc2n1 c1(C(=O)NCC(CC(=O)NCCc2cncnc2)O)nccc2cc[nH]c12 N1(C(C(C(C)C)O)=O)CC2CCC1C(N=c1nc(O)c3ccc(Cl)cc3[nH]1)C2 C(=O)(CS(=O)(=O)CC)N1CCC(N(C(=O)Cc2cccc(COC)c2)CCC)C1 c1(C(C(=O)NC(C2CN(C(CCC#C)=O)C2)C)C)ccc(N)cc1 Cc1nc(N2CC3CN(C(=O)Nc4cccc(Cl)c4)CC23)ncc1F CCC(CNC(=O)CNC(=O)CNC(C1(OC)CCOCC1)=O)CCO c1(C(=O)NCCC2CN(C(C34CC(F)(C3)C4)=O)C2)c(Br)nc2n1CCC2 N1(C(c2cc(C)sn2)=O)CCCC(NC(c2ccccc2Cl)=O)C1 CCC(C)C(C)CNC(=O)C(N1CCC(CNC(=O)Cc2ccccc2)CC1)=O CCCCCC(C)CC(=O)NC1(C(=O)NCCN(C(C)CC)C)CCN(C)C1 C1(C)(CNC(CC=C)=O)CC(F)(F)CN1C(c1cccc(C(N)=O)n1)=O C(C(C)N=c1ccnc(C(F)(F)F)[nH]1)NC(C(C)NC(c1ccccc1)=O)=O CCC(C(c1nnnn1C1COC1)NCc1nnnn1C)=Cc1ccsc1 C1(NC(C2CC2C2CC2)=O)CN(C(c2cc(-c3ccc(F)cc3)no2)=O)CC1O C(=O)(CCC(F)(F)C(F)F)NC1CC(CCn2cc(C3CCC(=O)NC3)nn2)C1 C(=O)(C1=C(C)CCOC1)NCC(CCC)NC(=O)C(=Cc1ccc(F)cc1)C Cc1cccc(C(O)C(=O)NC(C)CCCNC(=O)C(C)C(C)C)c1 CCCCCC(CC)C(=O)NCCC1CN(C(c2ncn(C)c2C)=O)CCO1 C1(C(N2C3CC(OC)C3CC2)=O)CCCCCCN1C(=O)CC1CCCOCC1 N1(C(N2C3CCC(C3)C2c2ccccc2)=O)CCCc2c(Br)cccc21 C1(NC(c2sccc2F)=O)CCC(C(=O)NOCCN(C)C)C1 N1(C(CCCC#C)=O)CC(CNC(=O)COCc2scnc2C)CCC1C c1(C(=O)NCC(CC=C)NC(c2cnc(C3CC3)o2)=O)nccc(Cl)c1Cl CCCCCC(CCCCC)CC(=O)NC(CN(C)C(c1occc1Cl)=O)CC N(C1CCOc2cc(OC)ccc21)C(=O)NCC(Cc1ccccc1)OC C12(C(N(CCN(C(C3(NC(C)C)CC3)=O)C)C)=O)CCCCC1C2(F)F CCC(CN(C)C)C(=O)NCC1CCN(C(=O)COc2ccc(F)nc2)C1 Cc1ccc(NC2CC2)c(C(=O)NCC2CCN(C(=O)CC(C)C(C)C)C2)c1 N1(C(c2ncc(C)nc2)=O)CCC(NC(=O)CCC2(C)CC2(F)F)CC1C CC1CCCc2cc(C(=O)NCCC3CCCN(C(C4CC4(F)F)=O)C3)nn21 C12(CNC(C3C(C)C3)=O)CN(C(=O)C(c3ccccc3Cl)O)CC(F)(C1)C2 O=C(CCC(F)(F)C(F)F)Nc1ccc(F)cc1Br N1(C(CCNC(c2ccc(C)nc2)=O)=O)CCCC2CN(C)CC12 C(=O)(CCCS(C)(=O)=O)NCCN(C)C(C1(C#N)CCC(=O)CC1)=O c1(CC)cc(=NC(=O)CC2CCCN(C(=O)C(CO)OC)CC2)[nH]n1C n1(C(C)C(=O)NC2(CCO)CC2)cc(CC2CC2)nn1 C#Cc1cccc(CNC(N2CCC(c3ccc(F)cc3)C2(C)C)=O)c1 N1(C(CN2CC(CC)C2)=O)CC(N(C)C(c2[nH]c(C)cc2C)=O)C2(CC2)C1 CCC(F)(F)CCNC(=O)CCN(C(=O)CCc1ccoc1)C1CC1 c1(CC(C)NC(=O)Nc2c(OC)cc(Cl)nc2)c[nH]c2ccc(OC)cc12 N1(C(Cn2ncc(C)c2)=O)CCC(F)(CNC(C2CC(C)OC2=O)=O)CC1 Cc1cc(=NC(=O)c2cc(C(=O)O)oc2C)[nH]n1-c1ccc(Cl)c(Cl)c1 c1(OC)ccc(C(O)C(N2CC(C(N)=O)(CNC(=O)COC3CCC3)C2)=O)cc1 c1(CCC(=O)NC(CC=C(C)C)(C)C)cccc(C(F)(F)F)c1 C1(C(=O)NCC2(CSC)CCC2)CCC(O)CN1C(c1cccc[n+]1[O-])=O Cc1nnc(O)c(C(N2CCC(NC(c3ccc(Cl)cc3O)=O)C2)=O)c1C C(C(O)CC(=O)N1CC(O)(CNC(c2cnco2)=O)C1)N(C)C Cc1nn(C)c(C)c1CC(=O)N(C)CC1(CNC(=O)CC(C)n2cccc2)CC1 c1(C(N2CCOC3CC23)C(=O)Nc2ccccc2Cl)cc(F)ccn1 N1(C(C)=O)CCOC(C(N2CCC(CCNC(c3ccc(Cl)cn3)=O)CC2)=O)C1 c1(OC)ccc(-c2nnc(SC(C)C)n2-c2ccc(SCCO)cc2)cc1 c1(C(=O)NC(CC)CNC(=O)Cc2csc(Cl)n2)cccc2occc12 c1(NC(N2CCCC(CN(c3ccc(Cl)cc3)C)C2)=O)cnn2cccnc12 C(C)(CN=c1[nH]cnc2c1COC2)OC.n12nccc1C(=O)NCC2 Cc1cc(C(=O)NCC(C)CN(C)C(c2cnc(C)cc2C)=O)cc(F)c1 N1(CCN(C(CCOC)=O)C)CCN(C(=O)CC2CC(C)=NO2)CC1 C1(C(=O)NC(c2cn(C)nn2)C(=O)NCC2CCCCS2)CCCCCCC1 N1(C(CCC2CC(NC(C(C(C)C)SCC)=O)C2)=O)CCN(C)C2(CCC2)C1 C(CC1=CCN(C(c2cc(CO)ccc2Cl)=O)CC1)NC(C(C)C1CCCO1)=O N1(C(C2CC3CCC2C3)C(=O)NCCC)CCC2(CC1)OCC(O)C2O C(C(N=[N+]=[N-])C(=O)N1CCCC1(C)c1ccccc1F)OCC N1(CC(=O)NCCN(C(C2(C)ON=C(C)C2)=O)C)C(=O)CN(C)C1=O n1(C(C)C)nc2c(cc1=O)CN(C(c1ccoc1Br)=O)CC2 C#Cc1ccc(F)c(C(N2CCC3C(NC(=O)C(C#N)(CC)CC)C3C2)=O)c1 C1(C)(N(C)C)CCCN(C(=O)CC=CCNC(=O)CC(C)(C)C2CC2)C1 C(=O)(C(C)(C)CC(=O)NC1CN(C(c2nc(C)oc2C)=O)CC1OC)OC CC1(C)CCC(NC(C23CCC(CC2)CC3)=O)C(CNC(C2(F)CC2)=O)C1 CC(CN=c1[nH]c2c(c(=NCC3CCCS3(=O)=O)[nH]1)COC2)n1cccn1 c1(C(=O)NC2CC(CCNC(Cc3cc(C)[nH]n3)=O)C2)ccc(C)c(C)c1F N1(C(CCC2C(C)C2)=O)CCC(C2(NC(C3CCNC(=O)C3)=O)CC2)CC1 c1(C(=O)NC2C=CCN(C(C(C)SC(F)(F)F)=O)C2)ccc2ccnn2c1 C1(C(=O)NC)CC1C1CCCCC1.C1(N)CC2CN(C(c3c(N)cccc3F)=O)CC12 c1(C(=O)NC(Cc2ccoc2)C(=O)NCC2CCCSC2)ccc[n+]([O-])c1 c1(N(C2CCN(C(CN(CC)CC)=O)C2)C)nc2cccc(C)c2o1 c1(C(=O)OCC(c2ccc(Cl)cc2)OC)cc2n(n1)CC(C)(C)CO2 C1(C(=O)NCC(CC)(CC)NC(CCC)=O)C2CCCCCCC12 c1(C(C)C)cnn(C)c1C(=O)NCC1CC(NC(=O)Cc2ccccc2Cl)C1 N1(C(C(C=CC)O)=O)CCC(F)(F)C(CNC(c2cc(F)c(F)cc2Cl)=O)C1 c1(CC(N2CCN(C(C3(Br)CCC3)=O)CC2)=O)ccc(F)cc1 N1(C(C(C)NC=O)=O)CCCC(CNC(c2cccc(I)c2)=O)C1 c1(C(N2CCC3(CCCCO3)C2)=O)cc(-c2cc[nH]n2)c2cc[nH]c2c1 n1(CCC(N2C(C)CCC(COC)C2)=O)c(=O)oc2ccccc12 N1(C(C(CCO)N(C)C)=O)CCC2(CCC2)C(NC(C2CC2F)=O)C1 C1(N=[N+]=[N-])(C(=O)NCC(NOCC)=O)CCN(C(c2nocc2Cl)=O)C1 Cc1ncc(C(=O)NCC2CN(C(C3CC3(c3ccccc3)C)=O)C2)c(=N)[nH]1 c1(OC)cccc(CC(=O)NC2CN(C(=O)Cn3nccn3)C2)c1Cl C1(C(N2CC(O)(CCNC(c3c(C)nc[nH]3)=O)C2)=O)OCC2CCCC1C2 c1(CNC(CC(=O)NC)C2CCCC2)coc2ccc(Br)cc2c1=O Cc1cc(C(=O)NCCCCN(C(=O)CS(N)(=O)=O)C)c2ccc(F)cc2n1 c1(Cn2cc(CNC3CCCC(C(=O)O)C3)nn2)cccc(F)c1 c1(CC)cc(OC)cc(C(=O)NC2CC(CNC(=O)COC3CC3)C2(C)C)c1 C1(NC(C=CCCC)=O)CN(C(=O)CSc2ccccc2)C2CCCC12 CCC(C)C(O)C(=O)NC1CCN(C(=O)COC2CCN(C)CC2)C(C2CC2)C1 C1(C(N2CC(F)(CF)C2)=O)(NC(C)=O)CCc2cc(Br)ccc2C1 C1(CCC)CN(C(c2cccc(OCC)n2)=O)CCN1C(C1CCCC1C)=O N1(C(COCCNC(C(C(CC)(C)C)O)=O)=O)CC(C2=NOC(C)C2)C1 N1(C(C(C)OCCC=C)=O)CCC(C)C(NC(=O)CC2CCC=CCC2)C1 c1(CCC(C)NC(N(CCCC)CC)=O)cccc(C)c1 C1(CNC(COC(CC)C)=O)C2CCC1CN(C(c1c(C)cc(C)cc1C)=O)C2 c1(N2CCCC(CNC(c3cnc4ncccn34)=O)C2)nc2c(F)cccc2o1 C12(C(=O)NC3C(CNC(c4ccc(OC)o4)=O)C3)CC3CC1C2C3O c1(C(C(=O)NC(C(C)NC(C2(C(N)=O)CCC2)=O)C)C)ccc(Cl)cc1 CC1CCN(C(C2(C(F)(F)F)CCC2)=O)CC1CNC(c1nc(O)[nH]c(=O)n1)=O CN1CC(=O)N(CC(=O)OC2(C(F)(F)F)CC(F)C2)C1=O C(c1ccnc2ccccc12)=CC(=O)N(CCNC(C1CC(C)C1(C)C)=O)C C1(F)(CNC(CC2(C)CC2(Cl)Cl)=O)CCCN(C(C2(C(F)F)CCCO2)=O)CC1 C(C(C)(CO)NC(=O)C(C)n1ccnn1)NC(C(C)NC(N)=O)=O c1(N(CCCC(C)O)C)nc(=NCc2ncccn2)[nH]c2ccc(Cl)cc12 c1(C(=O)NCCC(C)N(C(=O)CC2CCOC2)C)cc(C(F)F)ccc1F c1(C(=O)NCC(C)(CO)NC(C23CCC2C3)=O)ccccc1Br c1(C(=O)NCC(CC=C)NC(C2CC(OC)C(OC)C2)=O)c(F)ccc(Cl)c1F c1(C(N2CCC(CCNC(C(F)=CC)=O)C2)=O)oc2ccccc2c1CS(C)=O CC(C)CC(C(=O)NC1CC(CN2CCCC2)C1)NC(=O)C(C)(C)C C1(C(N2C(C(N(CC(O)C3CCC3)C)=O)CC=CC2)=O)CC2CCC1CC2 CC1CN(C(C2CC(F)(CO)C2)=O)C(C)CN1C(=O)CCc1ccon1 c1(C(=O)NC(c2cc(C(N3CCC3)=O)n[nH]2)C)ccncc1.C12CC1NC2 C1(C(=O)NC2CCC(CC)CC2)CCC(C)N(C(=O)CSCC(F)(F)F)C1 c1(CN(C(CN(C(c2cc(CC)no2)=O)C2CC2)=O)C)ccncc1C C1(CN(C)C(C2(F)CCCOC2)=O)CCC(CNC(=O)Cc2ncc(Cl)s2)CC1 N1(CC(=O)N(CC(C)NC(C2CCSC2)=O)C)C(=O)CCC1=O c1(C(N2CCN(C(=O)C=C(Cl)Cl)C(CCO)C2)=O)coc2c(F)cccc12 N1(C(c2cc(CC)n(C)n2)=O)CCC2(CC1)CC(NC(=O)CCC(F)F)CO2 c1(C(=O)NC2CC(NC(C(CC)(C)F)=O)C2)ccc(-n2cccn2)cc1Cl N1(C(c2occc2Br)=O)CC2CN(S(=O)(=O)Cc3ccc(Br)cc3)CC12 c1(NC(=O)NC(C(=O)NCC2CC2)Cc2ccccc2)cc(Cl)cnc1O CC1CCC(C)(C(N2CCC(C(O)CNC(=O)CCc3ncc[nH]3)CC2)=O)C1 C#CC1(CNC(=O)CC(C)CNC(c2ccns2)=O)CCOCC1 c1(C(N2CC(NC(C3C(COC)C3)=O)C2)=O)ccc(-c2nnc(S)o2)cc1 N1(C(C(C)CC(C)(C)O)=O)CCCc2cc(N3CCNC3=O)ccc21 C=C1CC(C(=O)OC(C)(C)C)(CNC(=O)C(C)NCC2(F)CC2)C1 C1(F)(CNC(C2C(OC)CC2)=O)CC(CNC(c2ncoc2C(C)(C)C)=O)C1 CC1(C)C(C)(C)C1(F)C(N1CCC(OCC(N2CCC(C)(C)C2)=O)C1)=O Fc1ccc(C(C(F)F)NC2CC3CC2CC3c2ccccc2)c(Cl)c1 c1(CCC)occc1C(=O)NC1CC1NC(=O)CCNC(=O)CO c1(CC)nc(C(=O)NCC(CC2CCCO2)OC)c2n1CCCC2 c1(C(=O)NCC2(Nc3ncnc(CC)c3F)CCCC2)cnc(O)c([N+](=O)[O-])c1 CC(C)C(CC(=O)NCc1cc(Cl)ccn1)NC(=O)Cc1ccon1 C(C)(c1ccco1)=CC(=O)NCC1C(C=C)C1 N1(C(CC(CNC(C2CC(CC3CC3)C2)=O)O)=O)CCOCC12CC2 c1(OC)ncccc1C(=O)NC1(CF)CN(C(=O)CCn2ccnc2)C1 c1(OC)cc2cc(C(N3CC(NC(c4cc(OC)no4)=O)C3)=O)[nH]c2cc1OC c1(OC)cccc(C(CNC(c2cc[nH]n2)=O)NC(C2C(F)(F)C23CC3)=O)c1 C1(NC(C2CC(OC)C2)=O)CC2CCC1N2C(=O)Cn1cnnn1 c1(C(=O)NCC2(NC(C3C(=C)C3)=O)CCOCC2)cc(S(N)(=O)=O)ccc1O c1(C(N2C(CNC(Cc3nnc(C)s3)=O)CC2)=O)nc(C)sc1C C1(OCC)CCCC(C(N2CCN(C3(C)CC3)CC2)=O)C1.c12ocnc1C(=O)N2 CC(O)(CNC(c1occc1CNC(C1COCC1C(N)=O)=O)=O)CO C1(CNC(c2ccoc2)=O)CN(C(=O)CCCn2ccnc2)CC12CC2 c1(C(=O)NCC2(F)CC(COC)C2)cnccc1OC.C12CC1C(=O)NC2 C1(O)(CCCNC(=O)CCOC2CCOC2)CN(C(=O)COCCN(C)C)C1 C1(CN(CCCCOC(C)C)C)CC[Si](C)(C)C1 N1(C(c2csnc2F)=O)CCC(C(O)C(F)F)CC1 c1(C(=O)NC2C(C(C)C)N(C(=O)C=CBr)CC2)ccc2c(c1)C=CS2(=O)=O CN1CCN(C(C2CCNC2=O)=O)CC1CNC(=O)CC(F)(F)Cl c1(C(=O)OC)cc(Cl)c(NC2(CCNC(C3CC(=O)N(C)C3)=O)CCC2)nc1C N1(C(C=CC=CCCCCC)=O)CCC(C)(CNC(c2ccnc(C)c2)=O)C1 C1(C(=O)NCC(CNC(c2c(C)noc2)=O)O)Nc2ccccc2C1(C)C Cc1cc(CC(=O)NC2CCC(NC(C34CC(C)(C3)OC4C)=O)C2)cc(F)c1 c1(C(=O)OCC)cnc2sncc2c1NC1COC2OCCC12 c1(NC(C2(C)CCN(C(C(C)=O)=O)CC2)=O)cn2cccc(Br)c2n1 N1(C(C(C)=C(C)C)=O)CCCCC1CN(C)C(C1C(Cl)(Cl)C12CC2)=O N1(C(c2cc(OC)no2)=O)CC2CCCC1C2CO N1(C(COC(C)=O)=O)CCCC(C)(C(=O)NCC(c2ccccn2)O)C1 N1(C(C(CC)CC)=O)CCN(C(=O)CC(O)C2CCCC2)C(CC(F)(F)F)C1 C(c1ccc(Br)nc1)=CC(=O)Nc1c(C(=O)OC)nn(C)c1 CCC(C(=O)NCc1cn(C2CN(C(c3cc(Cl)n[nH]3)=O)C2)nn1)OC C=CCCC(C)N=c1[nH]c(=NCC2(C)CC2(F)F)[nH]c2cc[nH]c12 C1(C(C)(C)C)CCc2sc(C(=O)NCC3CCN3C(=O)CCCC(N)=O)cc2C1 c1(CC)nc(C)[nH]c1C(=O)NC(C)CN(C)C(c1n[nH]c(C)c1Cl)=O C1(CC(=O)N(C2CCOC2)C)CC(F)CN1C(=O)CC1CCOC1 C(=O)(CS(=O)(=O)C1CCCC1)NC1CCN(C(c2cc(OC)n[nH]2)=O)C1(C)C n1(CC(=O)NC2(CNC(C(C=C)(C)CC)=O)CCOC2)nc2ccccn2c1=O Cc1cc(N(C(=O)CC(O)C2CCCC2)CCOC(=O)OC)n(Cc2ccco2)n1 C1(C(=O)NCC#C)CN(C(C2CCC(=O)C2)=O)CC1CCC c1(CC)conc1CC(=O)NCCC(C)N(C(=O)C=CC(C)(C)C)C c1(COC(CC2C(CC)C2)=O)ccn2cncc2c1 c1(C(N(CC(CC)NC(=O)C2=CC(C)(CC)C2)C)=O)cnc2n1CCCC2 c1(C(=O)NCCCN(C(C(C)N(CC)CC)=O)CC)ccnc2c(F)cccc12 c1(OC)nc(C)ccc1C(=O)NCC1(C)CCCN(C(=O)C(C)CC2CC2)C1 c1(C(=O)NC(C2CN(C(C3CCOC3)=O)C2)C)cncc(-n2cccn2)n1 c1(C(=O)NCC2(NC(C34CC(C)(C3)C4)=O)C(C)CCCC2)ccc2nccn2n1 N1(C(C2C(C(=O)OC)C2)=O)CC2CC1CC2CNC(=O)CSc1cnn(C)c1 N1(C(c2cc(C)nc(C)c2)=O)CC2(CCCC2)C1C(=O)NCC1CCC(C)C1 C1(C(N2C(C(C)(C)NC(c3n(CC)cnn3)=O)CCC2)=O)CCC(F)(F)C1 N1(C(C2C(C)(C)S(=O)(=O)C2)=O)CC2(COC(CNC(c3cnn[nH]3)=O)C2)C1 C1(OC)CC(NC(C2CC(O)C2)=O)CN(C(=O)C=CC2CCOC2)C1 c1(C(=O)NC2(CCNC(C34CCC(OC)C3C4)=O)CCCC2)cc(N)nc(Cl)c1 N1(C(C2CC=C(C)CC2)=O)CCN(C(C)=O)C(C)C1 N1(C(CC(=C)I)=O)CC(C)(C)C1Cn1cc(-c2cnc(C(C)C)o2)nn1 CCCCCCCCC(=O)NC12CCC(C1)N(C(c1ccc(C(C)(C)C)s1)=O)C2 c1(C(N2CCC(C)C(CNC(c3nc(Cl)cs3)=O)C2)=O)ccnc2cc[nH]c12 C12(C(=O)NC3C(CNC(c4cc5cccn5cn4)=O)CC3)C(=O)C3CCC1C2C3 C12(C(=O)NCCOCCN(C(C3C(C)C3)=O)C)CC(C)(C1)OC21CCC1 CCCCCCCC(C(=O)NCCCOC)N(C1CCN(CC(C)C)CC1)C CN1CCN(C)C(CNC(=O)C2=CCC(NC(=O)C=CC3CCCC3)C2)C1 C1(C)(C(=O)NC(c2ccc(Cl)cc2)C(C)C)CCN(C(c2cc[nH]c2)=O)C1 CC(C)C(CNC(=O)C(C1CCOCC1)C)C(=O)NCCN=S(C)(C)=O c1(CC(=O)N(CCN(C)C)Cc2nnn(C)n2)cnc(C(F)(F)F)nc1O N1(C(C=C(C)C)=O)CCC(NC(=O)CC2CCC(=O)N2)C(O)C1 Cn1ccc2c(C(=O)NC34CC3CN(C(=O)CCC3CCOC3)C4)[nH]cc2c1=O c1(C(=O)NCCNC(c2cnc(C(=O)OC)s2)=O)ccc(OC)cc1Cl N1(C(CCC(C)Oc2ccccc2Br)=O)CC(C)OC(C)C1 C1(C(=O)OC)(CNC(=O)C(=O)NCC(C)(C)CC2CCCCC2)CCOCC1 c1(Cc2nn(-c3c(C)cccc3)c(COCC3CC3)n2)c(F)cccc1F N1(C(CC(C)CF)=O)CC2CN(C(c3nocc3C(C)(C)C)=O)CC2C1 N1(C(CCCC#C)=O)CCCC(NC(c2ccc(-n3cnnn3)cn2)=O)C1C CCCC(C(=O)NCC1CC(NC(C2CC2C2CC2)=O)C1)N(C)C c1(C(=O)NCCSCC(=O)NCC(C=C)O)cncc(C#N)c1 c1(C(=O)NC2C(OC)CN(C(C3C(C=C)C3)=O)C2)noc2c1CCCC2 c1(OC)ccc(COC2CCN(c3ncnc(=N)[nH]3)C2)cc1 CC(=O)CCC(=O)NCC(C)CNC(c1cncc(Br)c1)=O C12(NC(=O)C(O)C3CCC3)CCCC1(F)CN(C(=O)C=CC1CCCCCC1)C2 c1(C(C(=O)NCC(CC=C)NC(C23CCCC2C3(F)F)=O)=O)cc(Cl)cc(Cl)c1 CC(C)C(C(=O)N1CCC(NC(C2CC=CC2)=O)C1)c1ccc(F)cc1 c1(CN2C(NC(=O)Oc3ccc(OCC)cc3)CC3CC32)c(F)cncc1Br.O N1(C(Cn2c(C)ncc2)=O)CCC(CN(c2ncccn2)C)CC1 c1(OC)cnc(C(=O)N(CC(C)N(C(=O)CCN2CCOCC2)C)C)cn1 CCCC(CC)CC(=O)N(C(CNC(=O)C(=O)NCC)CC)C c1(C(N(CCNC(=O)C(F)OC(F)(F)F)CC)=O)nnn2c1COCC2 Cc1ccc(Br)cc1NC(C1(F)CCN(C(c2cccc(F)c2)=O)C1)=O C1(C(C)NC(C=CCCC)=O)CCCCN1C(=O)CCNC(=O)CO C1(CNC(C(CCC)OCC)=O)CCN(C(=O)CC(C)O)C12CCC2 Cc1cc(C(=O)NCCC2CC(NC(=O)CNC(=O)C(C)(C)C)C2)no1 N1(C(CC(C)CN(C)C)=O)C2CCC1C1CC1(NC(=O)CCc1nncn1C)C2 CC1CCCN(C(=O)CCS(N)(=O)=O)C1CCNC(C1CCN1C1CCCC1)=O C1(C(N(CC(C)C(=O)NCC2CCCN2C)C)=O)CC(=O)C12CCC2 CCCCC(CNC(C1(NC(=O)CC2CCC(C)CC2)CC(F)(F)C1)=O)CCC c1(C(=O)NC(CC=C)CNC(c2oc(C)nc2CC)=O)ccc(C)nc1NC Cc1nn(CC(C)C)c(C)c1CC(=O)NC(C)CCCNC(=O)CCC(F)F C(C)(CC(=O)NCC1CCCN1C(=O)C=Cc1ccsc1)(C(F)F)N(C)C c1(C=O)ncc(-c2cn(Cc3nnc(C)o3)nn2)o1.C(C)(=O)OC CCC(C)C(C)C(=O)NCC(C(C)(C)C)NC(C1CN(C)CC(C)O1)=O Cc1ccc(C(=O)NCCN(C)C(c2cc(C3CC3)[nH]n2)=O)c(=O)n1C N1(C(=O)CC(F)(F)F)CCC(C2CCN(C(=O)CCC(=O)c3ccc[nH]3)C2)C1 N1(C(CNC(C(CC)C)=O)=O)CC(NC(C2(C)COCCO2)=O)C(C)C1 c1(C(=O)NCCCOCCCNC(C2CCCO2)=O)cnn(C2CCCC2)c1 N1(C(C(=C(C)C2CC2)F)=O)CCCC1C(C)NC(=O)CCCNC(=O)NC(C)C C1(Cc2nccc3[nH]ccc23)COC2(CCNC2)C1.c1(SC)nccc(C2CC2)n1 C1(CN(C(COCC(=O)OC)=O)C)CCCN(C(=O)CCCNS(C)(=O)=O)C1 c1(C(=O)NCC2C3CC2N(C(=O)CC2CC2(Cl)Cl)C3)c[nH]c2ccc(F)cc12 C=CCCCC(C(=O)NCc1cc(O)ccc1F)NC(=O)CCOC1CC1 c1(C(C)C)nccc(C(N2CCC(NC(=O)CC3CCC(=O)NC3)CC2)=O)n1 O=C1NCC(C(=O)NCC2(c3cc(F)ccc3F)CCCC2)c2ccccc21 CC1CCCC=C1C(=O)N(CC(C)(C)CNC(c1cnc2ccoc2c1)=O)C CC(C(=O)NC1CN(C(c2cncn2C)=O)C2(CCC2)C1)C(F)(F)C(F)F C1(OC)CC(NC(c2ccoc2C)=O)CN(C(=O)CCc2ncccc2C)C1 C1(C(=O)NC(C=CC(=O)NCCOC(C)C)(C)C)CCN(C)C1 N1(C(CNC(=O)OC)=O)CCCC12CN(C(c1cnc(OC)cc1OC)=O)C2 c1(C(=O)NCC2C(CNC(C(CC)N(C)C)=O)C2)csc2ncnc(O)c12 N1(C(c2cncc([N+](=O)[O-])c2)=O)CCC2(CCN(C(c3cc(Cl)c(Cl)[nH]3)=O)C2)C1 C#Cc1cc(C(=O)NC2(C)CC(NC(=O)CSc3nccn3C)C2)cc(Br)c1 C1(CNC(C(CSC)(C)C)=O)COCCN(C(=O)CCN2CCCC2=O)C1 C1(C(=O)OCC(CCC)O)CC(c2ccc(Cl)cc2Cl)=NO1 C(=O)(N1CCCCCO1)C1(CCNC(c2cncc(C=C)c2)=O)CCCN1CC CCC(CC)CCC(C(=O)NC1CCC1)N1CC(CO)C(C2CC2)C1 c1(CNC(C2N(C(CNC(CCC)=O)=O)CSC2)=O)cccc(C)n1 N1(C(C=CC)=O)CCCC1C1CCCCN1C(=O)Cc1cc(C)ns1 N1(C(C2C=C(C)CS2)=O)CCC(NC(c2cc(C)nnc2O)=O)C(C)(C)C1 CN1C(=O)CSC1=CC(=O)NCC1CC(C)(C)CN1C(c1ccc([N+](=O)[O-])o1)=O C12(SCC(CNC(c3cc(C(C)C)[nH]n3)=O)C)CC1CN(C(=O)OC(C)(C)C)C2 C1(C(=O)NCC2CC(NC(CS(CC)=O)=O)C2)CCN(C2CC2)S1(=O)=O CC1(C)CC(NC(=O)CC(F)(F)C(F)F)CN(C(=O)CC2(O)CCC2)C1 c1(C(=O)NCC(CN(C(Cn2nc(C)c(Cl)c2C)=O)C)O)c(F)ccc(N)c1F c1(C(=O)NC2C(CNC(C3(C#C)CCC3)=O)CCC2)cc(S(N)(=O)=O)n(C)c1 c1(C(=O)NCC(CNC(C(C)CC2CCCCC2)=O)C)cccc2nc(S)oc12 Cc1nc(CC(=O)NC(C)(CNC(=O)C(C)CN(C)C)CO)c(Cl)s1 c1(NC(COc2cc(C)c(F)cc2)=O)ccc2c(cnn2C)c1 C1(NC(C(CCC)C)=O)CCN(C(c2ccc(C)nc2N)=O)CC(C)(C)C1 C1(NC(C(CCNC(C2CC(C)(CC)C2)=O)OC)=O)CN(C)C(C)(C)C1 C#Cc1cnc(C(=O)NCC(CCC)C(=O)N2CCC(C#CC)C2)c(C)c1 C(Cc1cn[nH]c1)(C(=O)NCCc1csc(C)n1)NC(C1C(C(=O)OC)C=C1)=O C(CCC(CO)NC(C1CC(=O)N(O)C1)=O)NC(Cc1ccc(C)s1)=O C1(C(=O)NC2(COC)CN(C(C3CC(C(C)C)=NO3)=O)C2)CCC(=O)N(C2CC2)C1 C(=O)(CC(O)C(C)C)NC(C(=O)NCCc1scc(C)n1)CCC1CCC1 C1(C(=O)NCCCOCCCCCO)CCC12CCOCC2.C1(=O)COCCN1 N1(C(C(CCC)C#N)=O)CC(NC(c2cc(OCC)n[nH]2)=O)C2(CCC2)C1 Cc1ccccc1NCC(=O)N(CC(C)N(C)C(c1cnncc1O)=O)C c1(OC)ccnc(N2CCC(CCNC(=O)C(C)Oc3ccccc3)C2)n1 CN1CCCCC(C(N2CC(O)(CCNC(=O)C(F)OC(F)(F)F)C2)=O)C1=O C1(NC(C2CCC(CNC(COCC=C)=O)CC2)=O)CC(C)OC(C)C1 c1(OC)c(NC(C)CCNC(c2ccc(Cl)nc2C)=O)ncnc1C CC1(C(=O)NC2CCC(NC(c3csc(C(F)(F)F)n3)=O)C2)CCNC1=O c1(C(=O)NCC(CNC(Cc2c(C)cc(O)cc2)=O)C)cccc(F)c1C#N c1(-c2c(C(=O)NCC(F)CNC(C3(F)CC=CCC3)=O)c[nH]n2)ccc(F)cc1 C(=O)(C(C)(C)C(=O)OC(C)(C)C)N(CCCNC(=O)CCC1CC(F)(F)C1)C C1(O)(CC(=O)NC2C(NC(C(N3C(SCC)CCC3)=O)=O)C2)CCCCC1 C1(CC)C(C(N2CCC(O)CC2)=O)CCN1C(c1ccc(CO)cc1)=O c1(OC)cc(C(=O)NCC2CN(C(=O)C3CC3)CC2O)cc2c(C)c(C)[nH]c12 C(=O)(C1SCCc2ccccc21)N1CCC(C)(NC(CC(=O)N(C)C)=O)C1 CC1CCCC1(C(=O)N(C)CCc1ncccn1)NC(=O)C(=C1CCCCC1)F C(=O)(CC1=CCN(C(=O)C(C)(F)F)CC1)N1CCCC(OC(C)C)C1 c1(C(=O)NC2CC(C)N(C(=O)C#CC(=O)N(C)C)CC2)cnc2n(c1=O)CCS2 CCCC(CNC(=O)CCCCN(C)C)C(=O)NC(c1nc(C)cs1)C c1(SC)nc(=NC2CN(C(=O)Cn3ncc(O)nc3=O)Cc3ccccc32)s[nH]1 N#CC1CN(C(=O)Cn2cc(-c3ccc(C4CCC4)cc3)nn2)CCO1 C(C)(CCC(=O)OC(C)(C)C)N(C)C(c1cc(Cl)ns1)=O c1(C(=O)NCC=C2CCN(C(C(c3ccncc3)C)=O)CC2)ccc(S(N)(=O)=O)o1 c1(OC)cc(C(=O)NCCCNC(=O)CCc2ccccc2O)c(F)cn1 C(C(N=c1[nH]c(NC2CN(C3CCC3)C2)nc2ncn(C)c12)C1CC1)OC C1(NC(c2cc(C)c(F)cc2)=O)CCC2CN(C(c3cnc(Cl)[nH]3)=O)CC2C1 CC1=NNC(=O)C1CCC(N1CC2CC2(CNC(c2[nH]c(C)nc2C)=O)C1)=O C(CC)(C(=O)NCCCn1cc(CN(C)C(C)=O)nn1)OCC Cc1ccc2c(c1)CC(C(=O)N(C(C)CCNC(c1ncc(F)cc1C)=O)C)S2 N1(C(c2cc(C)n(C(F)F)n2)=O)CCCC(C)(NC(=O)CCCN2CCCC2)C1 C1(NC(C2CC(CC)OCC2)=O)CCN(C(C2CC(C)(CC)C2)=O)CC12CCC2 c1(C(=O)NC(CN(C(C(CC#C)C)=O)C)C)cc2cccnc2nc1C1CC1 N1(C(C2C(C(N)=O)C2)=O)CC(NC(C23CCCC2C3)=O)C(n2cccn2)C1 C1(CC(=O)NCCCCn2cc(COCC(N)=O)nn2)CC(O)C1(C)C c1(C(N2C3C(CNC(C(c4cccnc4)OC)=O)C(C3)C2)=O)ccc(N)c(N)n1 c1(C(=O)NC(CC)CNC(c2ccnc(Cl)c2F)=O)ccc(Cl)c(F)c1N C12(C(=O)NC(C(C)F)C)CC1CCN2C(c1cnsc1)=O C(=O)(CC(O)C(C)(C)C)NCCOC1CCN(C(COC)=O)CC1.C(CN)O c1(CN2CCN(C(Cc3c(C)noc3C)=O)CC2)ccnc2ccccc12 c1(C(=O)NC(CNC(C2(C=C)CCC2)=O)CC)cccc2c1OC(F)(F)O2 c1(C(=O)NC2C(CC(NOC)=O)CCC2)cc(C#N)oc1C N1(C(c2n(CC)c(O)nc2)=O)CCC2(CC1)CC(NC(C1(C)CC1(F)F)=O)CO2 CC(=O)CCN=C(NCC(C1CCOCC1)(C)C)NC(c1cccc(Cl)n1)C C(=O)(C(CCF)NC(c1ncsc1C)=O)NC(CN(CCC)CC)C c1(CC)cccc(CC(N2CCOCC2CN(C)C(C2CN(C)CCO2)=O)=O)c1 C12(C(N3C(CC(C)C)CC3)=O)CC(CN1C(C1CCC(=O)O1)=O)C2 Cc1cc(=O)ccn1CC(=O)NC1C=CCN(C(C2CCS(=O)(=O)CC2)=O)C1 Cn1cc(C(N2CC(CNC(C3CCCCC3)=O)C(O)C2)=O)c2cc(F)ccc12 C1(CNC(C2(C)CC2)=O)CN(C(=O)COC(F)(F)C(F)(F)F)CC12CCOCC2 c1(C(N2C3C(NC(CCC#CC)=O)(CCC3)CC2)=O)ccc2c(c1)C(C)(C)CO2 N1(C(c2csc(Cl)n2)=O)CC2(CCN(C(c3cnn4cc[nH]c(=O)c34)=O)CC2)C1 C(CNC(C1(CC2CC2)CC1)=O)(C(C)C)NC(C=C(C)C(C)C)=O C1(NC(c2c(-c3ccc(C)s3)ocn2)=O)CN(C(=O)CC2CCCCO2)CC1C c1(C(=O)OC)ccc(NC(=O)NCc2cncc(OC)c2)c(Br)c1 CN1CCC(C(=O)NCC2C3CN(C(=O)C(F)(F)c4cncs4)CC23)C1=O C(CC(=O)N(C)CCN(C)CCO)(C(C)CC)NC(c1c(CC)n(C)nc1)=O CCCC(O)CC(=O)N1CCCC(NC(=O)CCCN(C)C)C1C C1(CCOC)CN(C(c2cc(C)cs2)=O)CCN1C(=O)CCC1CCCCC1 c1(C(N(CC(CNC(c2cn(CCC)nn2)=O)O)C)=O)cc(F)cc(F)c1OC c1(C(=O)NC2CC(N(C(c3c(C(C)C)nn(C)c3)=O)C)C2)csc2cncn12 C(=O)(C(C)CN(C)C(C1CCCCC1)=O)NC(C)C(N)=O Cc1c(NC(C2OCCC2NC(C2CCCCCN2C)=O)=O)cccc1CO C#Cc1cn(C)nc1C(=O)NCC1CC2CCC1CC2 c1(CC)cnoc1C(N1CCC(NC(c2csc(CCP(C)(C)=O)n2)=O)C1)=O c1(C(N(CCCN(C(=O)C(C2(O)CCCC2)F)C)C)=O)ccnnc1 Cc1ccc(C(=O)N(CCCCCCNC(=O)C(C)CN(C)C)C)c([N+](=O)[O-])c1 N1(C(C(CC)NC(N)=O)=O)CC(NC(c2ncc[nH]c2=O)=O)C(C(F)F)C1 C1(NC(C=CC)=O)CCCCC12CCN(C(c1cc(C(C)C)[nH]n1)=O)C2 N1(c2nc(C)cc(C)n2)CCOC2(CCC(NC(c3csnn3)=O)CC2)C1 c1(C(N(CC(CNC(CSCC)=O)C)C)=O)c(Cl)csc1Cl c12cccc(c1)Cc1cn-2nn1.CC1(C)OC1C(=O)NC1CCSC1 C1(NC(CC2C(C)CN(C(=O)CCCn3ccnn3)C2)=O)CCc2n[nH]cc2C1 c1(OCC)cccc(C(=O)NC(CNC(=O)C(=Cc2cccs2)C)CO)c1N C(c1ccccc1C#N)=CC(=O)NC1C(C)(CNC(C2(Cl)C(C)(C)C2)=O)CCC1 C1(C(N(C(C(=O)NCC(CCC)(C)C)(C)C2CC2)C)=O)CNC(=O)CC1C c1(-c2cn(CC3CN(C(CCN4C(C)CCCC4)=O)C3)nn2)cc(F)ncc1F c12c(Cl)nnc(Cl)c1C(=O)OC2.c1(OC)ccc(C)o1 c1(OC)cccc(C(C)NC(=O)NCC(C)(C)C(C)C)c1 C1(CC(=O)NCC(=O)OC(C)C)C2CCCC2N1C(C1CC12CC2)=O C=CCC(C)(C)CC(=O)NCC1(C(=O)N(C2CC(OC)C2)C)CCCCC1 c1(C(=O)NCC(CC(C)C)NC(C(C=C)O)=O)cnn2c(C(F)F)cc(C)nc12 C#Cc1cccc(C(N2CC(NC(=O)CSCC=C)C(F)(F)C2)=O)c1F CC(CC(=O)NCCCCCN(C)C(C12CCC(C1)C2)=O)C(F)(F)F c1(C(=O)NCCCCNC(c2c(C3C(C)C3)noc2)=O)cnn2c1CCCC2 C1(CNC(C(=O)N(CC(c2ccncc2)C)C2CC2)=O)CCCN1c1nccs1 N#CCCCCCC(=O)N1CCC(CCNC(=O)COc2ccc(F)c(F)c2)C1 Nc1c(C(=O)NC2CCC(NC(C34CCN(CC3)CC4)=O)CC2)ccc(Cl)c1F c1(CC(=O)NCC2C(NC(c3ccc(C)cn3)=O)C2)c[nH]c2ccccc12 C1(NC(C(C(CC)O)C)=O)CCC2(CC1)CN(C(=O)C(c1ccccn1)O)C2 c1(C(=O)NCC2CC2NC(c2ccnn2CC(F)(F)F)=O)nc(Cl)cs1 C1(N(C)C)CN(C(=O)CCc2cccc(F)c2)CC1CNC(=O)C(O)CN(C)C N1(C(c2ccc[n+]([O-])c2)=O)CCCC2(CCCN2C(c2cc3sccc3[nH]2)=O)C1 C(CCC(C(=O)N1CCC(O)(CO)CC1)NC(c1cc(Cl)no1)=O)OC c1(C(=O)NCC2CCN(C(C(CC)n3nccc3C)=O)C2)cccc(C)c1O C(CC1CC1)(CC(=O)NCCC1COC(C)(C)C1)NC(CC(=O)OCC)=O Cc1ccc(C(=O)NCC2(C)CN(C(=O)Cc3cnoc3)CCO2)c(O)n1 c1(NC2C3CN(C(C(N4CCOCC4)C)=O)CC32)ncc(Br)cc1[N+](=O)[O-] N1(C(c2cscn2)=O)CCC2CCCN(C(=O)Cn3cnc([N+](=O)[O-])c3)C2C1 c1(C(=O)NC(C2(O)CCN(C(Cc3c(C)nc(S)s3)=O)C2)C)ncc(Cl)cc1F N1(C(CSC(C)C)=O)CCCC2(CNC(c3ccc(Cl)nc3O)=O)CC12 N1(C(CNC2CCC(=O)NC2)=O)CCCC2(c3ccccc3)CC2C1 c1(C(=O)NCCCC(C)(C)NC(C(C(C)C)SCC)=O)ccc2c(c1)ncn2C c1(CNC(C)Cn2cc(CO)nn2)nnc(N2CCCC2)o1 c1(CC)cc(C(N2CC(CNC(=O)Cc3csc(C)c3)CC2(C)C)=O)cc(F)c1 N1(CCCC(=O)NC2CC(C)(CNC(C(C)CSC)=O)C2)C(=O)CCC1=O C1(NC(=O)CO)CC2CC(NC(=O)COc3cccc(Cl)c3Cl)C1C2 C(=O)(CC1=CCN(C(c2ccnnc2C)=O)CC1)NC(Cn1ncc(C)c1)C CC(C)(F)CCC(=O)NCC1CC(C(=O)NCCCCc2ccccc2)=NO1 CC(CC(N)=O)C(=O)NC1CC2CCC1N2C(c1ccc(C(F)(F)F)nc1)=O Cc1cccc([N+](=O)[O-])c1C(N1CC(c2ocnc2CNC(C2CC(F)C2)=O)C1)=O C1(NC(=O)OC(C)(C)C)CCCN(N2CCC(NC(c3ccccc3)=O)CC2)C1 CC(CCNC(=O)C=CC1CCCC1)CCNC(C12CCCC1(C(N)=O)C2)=O c1(SC(C)C(N2CCC23CN(C(C2(N(C)C)CC2)=O)C3)=O)nc2ccccc2s1 c1(CC)ccc(C(N2CCCC(NC(=O)Cc3sc(O)nc3O)CC2)=O)c(C)c1 C12(C(=O)NCC3(CO)CCN(C(c4cc(C)nn4C)=O)C3)CCC(CC1)C(C)O2 N1(CCC(=O)NC(C2(O)CN(C(=O)C(C)(C)C(N)=O)C2)C)CCCc2ccccc21 c1(NC)cncc(C(=O)NCCCCNC(C2(SC)CC(O)C2)=O)c1 c1(C(=O)O)ccc2c(c1)N(C(C1CC3C=CC1C31CC1)=O)CCC2 c1(C2(NC(N3C(c4ccc(C)o4)CCC3)=O)CC2)cccc(P(C)(C)=O)c1 n1(CC(N2CC3C(NC(C(COC)N(C)C)=O)(C3)C2)=O)ccc(=O)n(C)c1=O CCCCC(C(=O)N(CCC)CCN(C)C)NC(=O)CC1CCCCC1 N1(C(c2c(C)c(C(F)(F)F)n[nH]2)=O)CC(NC(c2cnc(O)s2)=O)CCC1C N1(C(C)C)CC2CC1CN2C(c1ccc(CNC(=O)CCC(C)N(C)C)o1)=O c1(CC(=O)NC2(CNC(CCc3nc(C)sc3)=O)CCC2)ccc(CO)cc1F c1(C(=O)NCC2CC(O)(CNC(C(CC)OCC)=O)C2)ccc(Cl)c(F)c1 C1(C(C)C)CN(C(c2cc(O)ccc2Cl)=O)CCN1C(c1ncn2c1CCC2)=O CC1(C)CC(C(=O)NCCOCC2CCC2)N(C(c2ccn(C3CC3)n2)=O)C1 CC(=O)CCCCC(=O)NC(Cn1cncn1)C(N1CCCCCC1)=O c1(CC(=O)NCC2CC(C(=O)NCCc3ccc[nH]3)C2)cnccn1 c1(OC)ccc2oc(C(N3CC(F)CC3CNC(=O)C(C)(C)SC)=O)cc2c1 c1(C(=O)NC(CNC(C2(CCCC)CCC2)=O)C)cccn2c(C)nnc12 C1(CC)(CC)CC(NC(c2ccc(C#N)cn2)=O)CN1C(c1ccc(SC)s1)=O C1(NC(C(N2CCCCC2)C)=O)CCCC(CNC(=O)CCOC2CCCC2)C1 N1(C(C=C(CCC)C)=O)CCC2(CCC(NC(C3(CF)CCC3)=O)CC2)C1 C1(NC(CC(C=C)C)=O)CC2CC(C1)CN(C(=O)C(C)(C)N1CCOCC1)C2 N1(C(CCC(=O)OC)=O)CCCC2(CCN(c3ncnc4occc34)CC2)C1 C1(C(C)CO)CCN(C(=O)CC2CCCN2C(C2CC3C=CC2C3)=O)CC1 C1(C(N(C)CCNC(c2ccco2)=O)=O)CCCCN1C(C1CCCOCC1)=O N1(C(c2c[nH]c(=NC)s2)=O)CCN(C(=O)Cc2occc2C)CC1C(C)C CCC(CCOC)C(=O)N1CCOCC1CCNC(c1ccc[n+]([O-])c1)=O c1(C(=O)NCC2C(NC(C=C(CC)C)=O)CCCC2)ccc(N(C)C)nc1C C1(CCNC(C(C)OCC#C)=O)(C(=O)N(C)Cc2nc[nH]n2)CCCC1 N(C(=NCc1ccccc1)N1CCCCC1)CC(C(=O)OC(C)(C)C)(F)F CC1CCC(C)C1NC(C1CC(NC(=O)CN2CCNC(=O)C2)CCO1)=O N1(C(C(CC2CCCC2)NC(C2CC2(F)F)=O)=O)CC2CC2(CO)C1 CCC(F)(F)CCNC(=O)C(CCNC(=O)C(C)n1cnnn1)OC C1(CC(=O)N(C(CC(=O)NC(C(C)C)CN(C)C)C)C)CCCCC1O c1(OC)cc(F)c(NC(=O)CC2(CNC(c3nc(C)c(C)s3)=O)CC2)cn1 C(=O)(C1=C(c2ccccc2)CCC1)N(CCNC(C1(C#N)CCCC1)=O)C1CC1 C(CC1=CCN(C(C2(C)CCC(C)(C)CC2)=O)CC1)NC(CSCC#C)=O C1(C(=O)NC2(COC)CN(C(C3CCCC3)=O)C2)CCC2(CCC2)CO1 C1(NC(=O)CSCc2ccccn2)CCN(C(c2cnc(O)nc2O)=O)CC1F C=CC(CCC)CC(=O)N1CC(OC)C(NC(c2n[nH]cc2C)=O)C1 n1(CC)ncc(C(=O)NCC2CC3CC3N2C(=O)CN2CCCCC2)c1Cl C1(C(=O)NC2(CF)CCN(C(Cc3c(C)ncs3)=O)C2)CC12CCS(=O)(=O)CC2 C1(CC(=O)NC2C(C(=O)NCCOCCC=C)CCC2)C(C)(C)C1(C)C C1(CNC(C(C)CN(C)C)=O)CCC2CN(C(c3cnncc3O)=O)CCC2C1 C1(F)(CNC(CC2(C)CC2)=O)CCN(C(C2(C)CCOC2)=O)C1 C1(F)(CNC(c2cc(O)nc(Cl)c2)=O)CCN(C(=O)COC(F)(F)F)CC1 c1(C(CC)OC(c2n[nH]cc2C(F)(F)F)=O)cc(Cl)cn1C CC1CCN(C(=O)C(Cl)=CCl)CC1NC(c1cc(CN2CCC(O)CC2)on1)=O c1(NC(C2CC(NC(c3ccc(CCC)cc3)=O)C2)C2CC2)c(O)cccc1F CON(CCC(=O)N(C)C)C(=O)C(F)C(C)C.C1CN1C N1(C(C2(O)C(C)(C)C2)=O)CC2(CCN(C(c3cnc4ccsc4c3)=O)C2)C1 c1(CC)ccc(Br)cc1C(=O)NCC1CC(NC(C2(C)CC=CCC2)=O)C1 c1(C(N2CCC(COC)(CNC(=O)CC(O)CN(C)C)C2)=O)c(C)ccnc1O C1(CC)(CC)CC(C(=O)NC2(C(=O)N(CC(C)C)C)CC2C)C1 C1(C(N2C3C(N(C)C(C4SCCCS4)=O)CC(C3)C2)=O)CCC2(CCOCC2)O1 N1(C(CNC(C)=O)=O)CC(C)CN(C(=O)CSCCc2ccccc2)CC1C N(C(=NCc1nocc1C(C)(C)C)N(C)Cc1ccccc1)C(COC)C1CC1 N1(C(c2c(C)nc(CC(C)C)s2)=O)CCN(C(=O)C#CC(C)C)C(C)C1 N1(CC(C2CCS(=O)(=O)C2)OC)CCCCC1CNC(=O)CCc1nccn1C c1(OC)ccc(-n2cc(CNS(=O)(=O)Cc3cccc(C)c3)nn2)cc1 C1(CNC(C(C)=C(C)C)=O)CC(C)CN(C(c2cnn(CCO)c2N)=O)C1 CC(O)C(F)(F)C(=O)N1CC2CC2(C(=O)NC2CCN3CCC2C3)C1 c1(CC(=O)NC2CN(C(C(CC(C)C)O)=O)CC2O)cnn2c1OCCC2 Cc1noc(C)c1NC(c1nnnn1CC1CCOCC1)c1nccs1 N1(C(CC(C(=O)OC)(C)C)=O)CCC2(CC1)C(NC(=O)CCF)CS(=O)(=O)N2C N1(C(c2c(C(C)C)oc(C)c2C)=O)CC(C)OC2(CCN(C(=O)C(F)F)CC2)C1 C#CCCCCCCCC(=O)N1CCCCC(NC(=O)CCC(=O)NCCC)C1 C1(CCOC)(C(=O)NCC(n2cc(CCCSC)nn2)C)SCCCS1 C(C(C)C(F)C(=O)NCCCOC1CC1)NC(C(C)=CC1CC1)=O c1(C(CNC(C=C(C)C(C)(C)C)=O)NC(=O)CN2CCOCC2)ccccc1F S(=O)(=O)(c1ccc(Br)cc1NCCC1CCOC1)NC(C)(C)Cc1cccnc1 C(C(C)(C)CCNC(C1CC1(C)C)=O)NC(Cc1nc(C(C)OCC)sc1)=O C1(CNC(C2CC(=C)C2)=O)CCN(c2nc(Br)ns2)CC1C N1(C(c2cn(C)c(=O)nc2O)=O)CCC(CNC(C23CC(C2)C3)=O)C(F)(F)CC1 C1(CC(N2CC(C(C)C)C2)=O)CCCN(C(=O)CCN=[N+]=[N-])CC1 c1(C(=O)NCCn2cc(-c3cnc(C(=O)OC)nc3)nn2)ncn2c1CCCC2 C1(C(F)F)CC2(CC(NCC(c3cccc(Cl)c3)O)C2)C1 C(=O)(CC(O)C(C)(C)C)N(C1CCCN(C(c2cccc(C3CC3)c2)=O)C1)C Cc1cc(CNC(C2CCN2C(c2ccc3c(c2)CC3)=O)=O)nnc1C C1(C(N2CCOCC(CNC(C3(C(F)F)CC3)=O)C2)=O)COC2COCC2O1 N1(C(C(n2cc(-c3cnc(C)n3C)nn2)C)=O)Cc2ccccc2C1 C1(CC(=O)NCCN(C)C(C23CC(CC(F)F)(C2)C3)=O)OCCCO1 CCCC(C(=O)NC1CCCC1CNC(=O)CCCC1CCOCC1)N(C)C c1(C(=O)NCC2N(C(C=CC=CCC)=O)C3CCC2C3)cnn2ncccc12 N1(C(C(C(C)O)(F)F)=O)CCCC12CCCN(C(=O)CC1CCC(C)(C)CO1)C2 C(C(C)N=c1cccc(S(=O)(=O)NC(c2ccc(F)cc2)C)[nH]1)SCCOC CC1(CNC(=O)CCC2(O)CN(C(=O)C(O)c3ccsc3)C2)CCOC1 Cc1noc(C(C)C)c1C(=O)NCC(C)(CO)NC(=O)CC1CC2CC2C1 N1(C(C(c2ccccc2)C)=O)CCCC2(CC(NC(C3CCC=CCC3)=O)C2)C1 N1(C(CC(=O)NCC)=O)CCC(C)(CC(N2CC(c3ccncc3)C2)=O)C1 C1(C(N2CCC(C)(CNC(C3CNC(=O)C3)=O)C2)=O)CC(c2ccccc2)=NO1 C1(NC(C2(NC(=O)CCc3ccsc3)CCCCC2)=O)CCC12CCCC2 C(=O)(C1CCc2cccnc21)NCC1N(C(C(C)NC(=O)C(C)(C)C)=O)CCC1 C1(C(=O)NCC(N2CCN(C(CC(C)CF)=O)CC2)=O)CCC2(CCOCC2)C1 c1(N2CCN(C)C(c3ccccc3OC(F)(F)F)C2)nc2cc(F)ccc2o1 N1(C(C)=O)CCN(C(=O)CCCNC(=O)C(C)(C)C)CCNCC1 C(C(=O)NNc1cccc(Br)c1)c1nnc(-c2cc(CC)on2)n1C N1(C(c2cc3oc(Br)cc3s2)=O)CCn2c(Cc3cncc(O)c3)nnc2C1 c1(-c2ncc(C(=O)Nc3c(OC)ccc(Br)n3)nc2)ccc2sc(C)nc2c1 C1(C(N(CC(=O)OCC)C)=O)CC12CC(NC(C1(C)CC1C)=O)C2 Cc1ccncc1NC1(c2nnnn2CCCC2CC2)CCCC1C CCCC(C(=O)N(C)CC1CCCCN1C(C1(SC)CC1)=O)NC(N)=O c1(C(N2CCCC2CNC(C2(N(C)C)CC2)=O)=O)nc(N2CCOCC2)ncc1Cl CC1(C(N2CCC(NC(c3csc(-c4cccnc4)n3)=O)C2)=O)COC(=O)C1 CC(F)(F)CCCC(=O)NC1CCCC12CN(C(C1CCC3(CCOC3)O1)=O)C2 CC1OCCC1(O)CNC(C1(N(C(=O)Cc2cccnn2)C)CC1)=O C(CC(C)(C)NC(C1CCC1n1ccnc1)=O)NC(C1C(CCOC)C1)=O C(=O)(C(CO)C(F)(F)F)NC1CC(C)(NC(=O)COCC(F)F)C1 C1(NC(C(c2c(C)n[nH]c2C)C)=O)CCC2CC1CN2C(c1cn(CC)nn1)=O CCC(O)C(C)(C)C(=O)N(CCNC(C1CCCN(c2nccs2)C1)=O)CC C1(c2c(OC)cc(F)c(F)c2)NC(=O)N(CCF)C2=C1C(=O)NC21CCCCCC1 CCCC(C)=CC(=O)NCC1CC(NC(=O)C(C)C2CCCC2)C1 N1(C(CC2(C)CCN(C(c3cncc(C=C)c3)=O)C2)=O)CC2CCCC(O)C2C1 N1(C(c2c(CC)c[nH]n2)=O)CCN(C(c2cnc(C(C)(C)C)o2)=O)C(C(C)C)C1 c1(OC(C(N2C3C(NC(C=C(C)Cl)=O)CC(C3)C2)=O)C)cccc2ccccc12 C(=O)(CCN=c1[nH]ccs1)N1CC2C(NC(c3c(C)con3)=O)(CCC2)C1 CCCC(C(=O)NC1(c2cn(CCNC(=O)C(C)C)nn2)CC(F)(F)C1)C(C)C C1(C(N(C(=O)C(=O)C(C)(C)C)C2C(CC)CCCC2)=O)CCCC12CCOCC2 c1(CNC(c2n(CCC)nnn2)c2ncc(CSC)s2)c(F)c(F)cc(F)c1F C1(C(N2C3C(NC(c4cc(CC)ncc4)=O)C(C3)C2)=O)CCC=CCCC1 c1(C(=O)NC2C3(CN(C(C(C#C)(C)C)=O)C3)CCC2)cccc2nc(C)cnc12 c1(C(=O)NC(C)CN(C(=O)Cc2cc[nH]c2)C)ccc(CN2CCCCC2)cc1 S(=O)(=O)(CCCC(=O)OC)N(CC)Cc1occc1C.C1(=O)CO1 N1(C(c2c(OC)nccc2)=O)CCC(C2CC2)C1C(=O)NCC(C)(C)C(C)(F)F C=CC(CCC)CC(=O)NCCC1(C)CCN(C(=O)CNC(C2CCC2)=O)C1 C(=O)(C1=NOC2(CCOC2)C1)NCCC1N(C(CCCN(C)C)=O)CCSC1 C(C)(N=c1ccnc(NCC2(C)CCCO2)[nH]1)c1c(OC)nccc1 c1(C(=O)NCC2N(C(CC=CCC)=O)CC2)cnc(C(C)(F)F)s1 C1(OC(=N)O)CCN(C(=O)C(F)CC2CN(C(C34COCC3C4)=O)C2)CC1 c1(C(=O)NC2C3CCC2N(C(=O)COc2ccsn2)C3)cc2nn[nH]c2cc1F C1(C(=O)NOCC=CCl)(NC(c2coc(C3CC3)c2)=O)CC(F)(F)C1 c1(OC2(CC(=O)NCC(C)CN(C(=O)CC3(O)CC3)C)CC2)ccccc1 c1(-c2cc(CN3CC(CC)OCC3)[nH]n2)cccc2c1OCO2 C1(C(=O)NC2C3CCN(C(CCc4c(C)n(C)nc4)=O)C32)CC(C)(C)OC1(C)C C1(NC(CN(C(C)C)C)=O)CN(C(c2ncccc2O)=O)CC1CO C(=O)(CCCC(F)(F)F)NCC1C(CNC(COc2c(C(N)=O)cccc2)=O)C1 C(=O)(C1=CCc2ccccc21)N1CC(C)OC(CCNC(c2cn(C)nn2)=O)C1 c1(C(C(=O)NC(CC)C)N(C)Cc2ncc(Br)s2)cc(OC)c(Cl)cc1F S(=O)(=O)(c1cccc(I)c1)NCc1n(C)c2c(n1)CCCC2 CCCC(CC)C(=O)NC(C)(C)C(C)NC(c1cc[nH]n1)=O C1(NC(C(CCC)O)=O)CN(C(=O)CCOCC(F)(F)C(F)F)C2(CCC2)C1 c1(C(=O)NCC(CO)NC(CCC#N)=O)cccc(C2CC2)c1Cl C1(NC(C(C)SCCCC)=O)CC2CCC1N2C(c1nccc(C)n1)=O CC1CC(NC(C2CCOCC2(C)C)=O)CN(C(=O)C=CCO)C1 c1(C(=O)NCC2(CNC(c3c(C)coc3C)=O)CC2)cc(F)c(Br)c(F)c1 C1(NC(C=CCOC)=O)CCC(C(=O)NCC2CC(F)(F)C2)CC1 C(=O)(CC1=CCN(C)CC1)NC(CC(C)C)CC(=O)N1CCC(N(C)C)CC1 C(N=c1[nH]c(=NCCOCC2CCOC2)c2sccc2[nH]1)c1cccnc1 c1(OC)c(C(=O)NC2CC3CC2CN3C(=O)C(C(C)C)NC=O)cc(F)cc1F N1(C(c2conc2CC2CCCC2)=O)CCC2(CC(C(N3CCC3CF)=O)C2)C1 CC(C)CC(Cc1ccccc1)C(=O)N1CC2C(Cc3nn[nH]n3)C2C1 C1(CC#N)CN(Cc2ccc(C(F)(F)F)cc2)CCN1C(=O)CC1CCOCC1 C1(CC(N2CCC2CO)=O)C2CN(C(=O)CC3CCC3)CC12 c1(C(c2nnnn2C2COC2)NC(CCC)C2CCC2)cccc(F)n1.CO C=CC(C)(C)CC(=O)N1CC(CNC(c2cnc(O)c(C)c2)=O)C(C)C1 N1(C(C(C(=C)C)(C)C)=O)CC2CCCC(C1)N2C(c1cc(Cl)c(F)cc1O)=O CC1CN(C(C2(F)CCCC2)=O)CC(C)N(C(=O)COc2cc(F)ccc2F)C1 N1(CC(=O)NC2CC(CCNC(C(COC)C)=O)C2)CCC(C)(C)C1 c1(C(=O)NCCN(CC(C)O)C(=O)CC2CCCC(=O)N2)cnc(O)n1C N1(C(C2COCC(C)O2)=O)CCC2(CC2C(=O)NCCc2ncc[nH]2)C1 c1(OCC(=O)OCC)ccc(S(=O)(=O)Cc2cccnc2)nc1 C(=O)(CCS(C)=O)N(C(C)C)CCNC(c1cccc(N(C2CCCC2)C)c1)=O C1(CN(C(=O)Cc2cncnc2)C)CN(C(c2coc(Br)c2)=O)CC12CC2 C(=O)(C(CNC(c1nnc(S)n1C)=O)(CC)CC)NC(CCSCC)C c1(NC(C(C)NC(=O)CCc2ccccc2)=O)cc(F)ccc1Br N1(C(C2(C(=O)NC)CCC2)=O)CC=CC1CNC(C1CC1C(F)F)=O C1(C(=O)NCC2CCCC(NC(c3scc(OC)c3)=O)C2)CC1C1CC(F)(F)C1 c1(C(N2CCC(N(C(c3ncc(C)cc3F)=O)C)C2)=O)cc([N+](=O)[O-])nn1C c1(C(=O)O)cccc(S(=O)(=O)N2CC(F)(C(=O)Nc3ncc(Br)cc3O)C2)c1 c1(CC(=O)NC2CC(CNC(=O)Cn3cncn3)C2)cccc(F)c1 CC(C)S(=O)(=O)C(C)C(=O)NC(C)CNC(c1cc2nccc(Cl)c2s1)=O N1(C(CSCC(C)=O)=O)CCCN(C(=O)C=CC(c2ccccc2)=O)CC1 N1(C(c2cc(C)c(O)cc2)=O)CCCC1C1CCCCN1C(c1cc(Cl)ns1)=O C1(C(=O)NCCC2C(C)CN(C(=O)C3=CCCCO3)C2)CCn2c(O)nnc2C1 CCC(C(F)(F)F)NC(C1CCCC1NC(c1c[nH]c(=NC)o1)=O)=O N1(CC)CCCC2(CCN(C(c3ccccc3N3CCC(O)CC3)=O)C2)C1 C1(C)(C(N(C2CN(C(c3cc(C(O)C(F)(F)F)ccn3)=O)C2)C)=O)CC2CC2C1 CC1CC(NC(C2CC(O)C2)=O)CCN1C(=O)Cn1nnc(-c2cccs2)n1 c1(-n2cc(Cc3ccc(COC)c(F)c3)nn2)ccc(Br)cc1F N1(C(CCOCC#C)=O)CC(NC(=O)Cc2ccc(C)cc2F)CC(C)C1 CC1CCC(NC(=O)C(=O)N2CC(NC3(c4cccnc4)CCCC3)C2)C1 N1(C(C2CCN(C(C)=O)CC2)=O)CC2(CCN(C(=O)C#CC3CCCO3)C2)C1 C1(N(C(C=CCOCCOC)=O)C)CCN(C(=O)Cn2cccc2)C1 N1(C(C(C)(C)O)=O)CC2C3CCC(C(NC(c4ccc(F)c(CO)c4)=O)C3)C2C1 Cc1cnc(NC(c2c(F)cccc2I)=O)nc1C c1(CC)cc[nH]c1C(N1CCCC1C(N1CC(NCC)C1)=O)=O.C(C(N)=O)O C(=O)(CC(C)CC(=O)NC1CCC(C(=O)NCC(C)SC)C1)OC C1(C(N2CCN(C(c3ccsc3)=O)C(CO)C2)=O)CCOCC12CCC2 c1(C(=O)OCC)cc(Cl)cc([N+](=O)[O-])c1NC(=O)CCCSC Cn1nnc2c1CC(C(=O)NCC1CCCC1NC(=O)CC=C(Cl)Cl)CC2 N1(C(C23CCC(OC)(CC2)C3)=O)CCN(C(=O)CO)C2CCCCC12 N1(C(C2N(C(CNC(C3C(C)(C)C3)=O)=O)CC2)=O)CC(C)(O)C1 N1(C(c2c(C)scn2)=O)CCCC(CNC(c2cnn(C(C)(C)C)c2N)=O)C1 Cc1conc1CC(=O)NCCOC1CN(C(C2(Cl)CC2C(C)=O)=O)C1 C(=O)(CC(F)(F)C(F)F)NCC1CCCN(C(c2c(OC)nc(Cl)cc2)=O)CC1 N1(C(C(C)(C)OCC(F)(F)F)=O)CCC2(CC(NC(=O)CC=C(Cl)Cl)CO2)C1 N1(C(c2c(F)ccc(C)c2)=O)CCC2CC2(NC(c2ccc(F)s2)=O)CC1 C1(C(N2CCCC(CNC(C(C)(C)F)=O)CC2)=O)OCCOC12CCC2 c1(C(=O)NC2(CO)CN(C(C3(CCCC)CC3)=O)C2)cn(CCOC)nc1C C1(C2N(C(C(C)OCCN(C)C(C34CC(F)(C3)C4)=O)=O)CC2)CCCCC1 CCCCCC(C)CC(=O)NC1(COC)CN(C(=O)C(F)(F)c2ccccn2)C1 N1(C(c2cn(C)nc2C(F)(F)F)=O)CCC2(CCCC2C(=O)Nc2ccno2)C1 c1(-c2nnc(CN3CCC(C)(CC(=O)OC)CC3)n2C)cnc2[nH]nnc2c1 Cc1nc(C(N2CC3(NC(=O)CCC4CC4)CCC2C3)=O)c(C)n1C N1(C(c2cnn(CC)c2C)=O)CC(C2CCCN(C(=O)C(C)C(C)(C)C)C2)C1 C12(CCNC(c3occc3Cl)=O)CCC1CN(C(c1ccc[n+]([O-])c1)=O)C2 Cc1nc2cc(Cl)cc(C(=O)NCC3CCCN3C(=O)Cc3cncnc3)c2[nH]1 N1(CC(N2CCC(c3nc(C(=O)O)n[nH]3)CC2)=O)C(=O)C2C3CCC(O3)C2C1=O S(=O)(=O)(c1nccs1)NC1CC(CC(N2CCC(C#N)C2)=O)C1 N1(C(c2scc(C#N)c2)=O)CC(NC(C2CC2F)=O)CC12CCOCC2 C12(CNC(c3c(CC)ncs3)=O)CN(C(C3(C)CC(F)C3)=O)CC1CCO2 N1(C(C(C)(C)c2ccccn2)=O)CC(NC(c2cc(F)cs2)=O)C(O)C1 n1(CCCC)nc(C)c(C(N2CC(CNC(c3ccc(Cl)o3)=O)C2)=O)c1Cl Cc1ccc(C(N2CCC(N(C)C(c3cccn3C(C)C)=O)CC2)=O)c(F)c1 C(CC(C(C)(C)C)NC(=O)Cc1nnc(S)n1C)N(C(=O)C=Cc1cccs1)C C#CC1C(C(=O)N(C2CCN(C(=O)C(C)(O)CC)CC2)CC)C1(C)C C1(NC(c2cc(CCC)on2)=O)CN(C(c2cn(C)nc2C(C)C)=O)CCC1O c1(OC)nc(C)cnc1C(N1CCCC1c1cc(C)cc(C)c1)=O Cc1oc(Br)cc1C(=O)N(C)CCOCCCNC(=O)C(C)(F)F CCC(CC(C)C)C(=O)N(C)CCNC(C1CNC(=O)C(C)(C)C1)=O N1(C(c2c(C)onc2C2CC2)=O)CCC(NC(=O)CCS(C)=O)C2(CCC2)C1 c1(CC(=O)OCC2CCCN(C(=O)NCC(F)(F)F)C2)cc(Cl)c2c(c1)OCO2 C(F)(C(=O)NOCC(O)CO)C1(O)CN(C(C(C)C2CC2)=O)C1 CC1Oc2c(F)cccc2C1NCCC(C)(c1ccccc1)NC(=O)OC(C)(C)C C(=O)(C(C(C)NC(c1cnc(C)cc1C)=O)C(C)C)N(CC(=O)OCC)C O=C(CN=c1cc[nH]cc1)NCCCNC(=O)COc1ccc(Cl)c(F)c1 N1(C(c2c(CNC(=O)CCCF)nccc2)=O)CCCC12CCCC2 N1(C(C(=O)N(C2CC(O)C2(C)C)C)=O)CC(NC(=O)C2CC2)C(C)(C)C1 N1(C(C23CC(C(=O)OC)(C2)C3)=O)CC(NC(c2cccnc2)=O)C2(CCC2)C1 Cc1cc(-c2cn(CCC3CC3Cc3ccccc3)nn2)ccc1F c1(NC(CO)C2CCC2)cnc(Cl)cc1Cl c1(C(=O)NC2CC(C(C)NC(c3ccc(CCC)s3)=O)C2)cccc2ccoc12 C1(c2n(CCCC)nnn2)(NC(c2cc(F)ccc2C)CC)CCN(CC)CC1 c1(C(C(=O)NC(C)C)N(C(C)C(=O)OC)CC)cc(C(OC)OC)on1 C1(N(C(C(COC)C)=O)CC2CC2)CCN(C(=O)CC2CCNC(=O)C2)CC1 CC(C)C(C(=O)N(C1CCCN(C(=O)CC(C)(C)C)C1)C)N1CCCCC1 O=C(CN=c1ccnc(NCC2CCC3CC23)[nH]1)NCc1nc2ccccc2s1 N1(C(=O)CSCC2CCCC2)CCOC(c2cn(Cc3ccc(F)cc3)nn2)C1 N1(C(c2nc(Cc3c(C)cc(C)s3)sc2)C)CCc2cc(C#N)ccc2C1 C1(NC(C2CC(C#N)C2)=O)CN(C(C2CC2(Cl)Cl)=O)C2(CCCCC2)C1 C=C(C)C1OCCCC1C(=O)N(CCC(C(C)C)NC(=O)CCSCCCC)C c1(SC)c(C(=O)NC2CCCC(NC(=O)CNS(=O)(=O)N(C)C)C2)cnn1C N1(C(C2CCCC(C)C2)C(=O)Nc2cccc(OC)c2)CCC(O)C(C)C1 N1(C(CCCOC(C)=O)=O)CCn2ncc(CNC(=O)Cc3ccon3)c2C1 c1(CC(=O)NC2C(NC(C3(C#N)CCCC3)=O)CC2)cc(F)cc(F)c1 C1(NC(=O)C=Cc2cocn2)CC2CC(C1)N(C(C1(C3CCCCO3)CC1)=O)C2 C#CCC(CC(F)F)C(=O)N1CCC(C)(CNC(=O)CN2CC(=O)NC2=O)CC1 Cc1nc[nH]c(=NCC23CCCC2CN(C(=O)C=C2CCC2)C3)c1Br n1(C(C)C)cc(C(=O)NC(C)CNC(C2SCCN2C(=O)OC(C)(C)C)=O)nn1 C(=O)(C(CC(C)C)C(C)C)NC(CC#C)(C)C(=O)Nc1cccc(OC)c1 c1(C(=O)OC)cc(F)c(C)c(NC(c2nccc(C)c2Br)=O)c1F c1(C(N2CC(C)(NC(=O)Cc3cn[nH]c3)C2)=O)ccc(OCc2cscn2)cc1 N1(C(c2c(SC)cccn2)=O)CCN(C(C2CNC(=O)C2)=O)C(C)C1 C1(c2cccc(C(=O)OCC)c2)CCN(N2CCCN(CC)CC2)CC1 c1(CCn2c(COCC)nnc2N(C)Cc2cccc(F)c2)ccc(Br)cc1Cl N1(C(C2C(COC)CC2)=O)CCSCC1C(=O)N(C1COCC1O)C N1(C(c2cncc(C)n2)=O)CCC(n2cccn2)(C(N2CC(C)C2)=O)CC1 C12(CNC(CCCCOC)=O)CCCC1CN(C(C13CC4CC1C3C4)=O)C2 NC(=O)CCCC(=O)NCCN1CCN(C(c2ncncc2F)=O)CC1 CCC(CC(=O)N(CC(=O)NC1CCC1)CCOC)OCCC(=O)OC c1(C(N2CCC(C)C2CNC(c2ccc(F)o2)=O)=O)cc(C#N)ccc1Br O=C(C#CC1CCOC1)NC1CC2(C(=O)NCCc3cccs3)COC1C2 N1(C(CC2C(=O)OCC2)=O)CC23CCCC2(C1)CN(C(=O)Cc1ccsn1)C3 c1(C(=O)NC2CC3(C2)CN(C(C2CCCC2O)=O)C3)cc2c(Cl)cc(F)cc2[nH]1 C1(C(=O)NCC(CNC(C(C(C)C)OC)=O)S(C)(=O)=O)CCC2(CCCC2)C1 n1(C(C)C)cc(C(=O)NC(C2CN(C(c3cc(F)c[nH]3)=O)CCO2)C)ccc1=O CC(C)C(O)CC(=O)NC(C1(O)CN(C(=O)CC2(c3ccon3)CC2)C1)C Cc1cc(C)c(C(=O)NC2(CNC(=O)CC3COCCN3C)CCOC2)cc1C c1(C(N(CC(C)NC(C2(C)CC=CCO2)=O)C)=O)ccc(C2COC2)cc1 c1(C(=O)NC2CN(C(c3c(CC)n(C)nn3)=O)CC2(C)C)cc2n(n1)CC(F)C2 N1(C(c2cnc(C)n2C)=O)CCC(C(=O)NCCC(C)(O)C2CC2)=C(F)C1 N1(C(c2c(Cl)ccc(NC(C)=O)c2)=O)CCC(C)C(NC(=O)C(N)=O)C1C C(=O)(CCCC(=O)OC1CCCC1)N1C(C)CC(NC(CC(=O)NCC)=O)C1 Cc1cc(F)cc(C(N2CC(NC(C34CCCN(CC3)C4)=O)C2)=O)c1N C1(CC(=O)NCc2ccc(OC)s2)CN(C(c2nc(Cl)oc2C)=O)CC1C CC1(C)CN(C(=O)CC2(O)CC2)CCC1NC(C1COCCO1)=O C(c1cccc(O)c1)=CC(N1C(C)CC(CNC(Cc2cc(C)sc2)=O)C1)=O C1(NC(CC=CC)=O)CN(C(C2CCCC23CC3)=O)CC2(CC2)C1 CC1CCNCCC1N(C(C1CCC(=O)NC1)=O)CC1CCOCC1 C(=O)(CCCC(=O)NCC1CCC1NC(C1(C)CC(C)=NO1)=O)N(CCC)CCC c1(C(N2CC(NC(C3(C)ON=C(C)C3)=O)C2)=O)cncc2ccccc12 CC12CC(C(=O)NC3CC3NC(c3ncoc3-c3cccs3)=O)(C1)C2 c1(C(C(N2CCN(CCNC(=O)C(F)n3ccnc3)CC2)=O)O)ccc(F)cc1 N1(C(C2(NC(CC(COC)C)=O)CC(F)(F)C2)=O)CCNC(=O)CC1C C1(CC(=O)N(C2CCN(c3cccnn3)CC2)CCO)Cc2cc(Br)ccc2C1=O N1(C(C2N(CCC)CCC2)=O)CCC=CC1C(=O)N(C)Cc1ncnn1C C1(C(=O)NCC(CCC)NC(C(CC(=C)C)NC(C)=O)=O)CCn2cncc2C1 N1(C(=O)NCC(c2ccccc2)OC)CCC(NC2CCC2)C1 CC1CCCC(C(=O)NC2CN(C(c3ccc(F)c(F)c3)=O)CCC2C)CC1 C1(C(N2CCC(C(C)NC(c3nc(CC)[nH]n3)=O)C2)=O)CCCC2C1C2(F)F c1(NC(=O)NCC(CN(C)C)O)nc(Cl)sc1Cl CC1(C)CC(CNC(=O)C(C)(C)N2CCCC2)N(C(C23CCC(F)C2CC3)=O)C1 C(=O)(C#CC1CCOCC1)NC1(CCNC(c2c(C)nn(C)c2N)=O)CCCC1 c1(CSC)noc(CCC(=O)NCCNC(=O)C(C)CN2CCOCC2)n1 C(=O)(CS(=O)(=O)Cc1cccs1)NCC(CNC(C1(C)ON=C(C)C1)=O)(C)O C1(C(=O)OC)CCC(n2nnnc2C(C2(CC#N)CC2)NCC(C)(C)CO)C1 C1(NC(C(C)N(C(=O)CC2CCOCC2)C2CC2)=O)CCN(C2CC2)C1 CC1OCCC1(F)C(=O)NCc1cc(C(=O)NCC2=CCCCC2)ccn1 N1(C(=O)CC2COCCO2)CCC2(CC1)CCN(C(C1CC(C(F)F)C1)=O)C2 N1(C(C(=O)NC2CCN(C(=O)OC(C)(C)C)C2)=O)C(C(=O)O)CC2OCCC12 CC1(C)CC2(CC(c3nnnn3C(C)(C)C)(NCc3cnccc3Cl)C2)C1 Cc1cc(C(=O)OC(C)(C)C)c(Br)cc1F.C1(=O)C(c2cscn2)NC(=O)N1 c1(CC(=O)NCC2(CNC(C)=O)CCC2)cccc(N2CCOCC2)c1 N1(C(C(CCC)CC)=O)CCc2[nH]nc(CNC(C3CC4CC4C3)=O)c2C1 c1(C(N2C3C(NC(c4c(C)cnn4C)=O)CC(C3)C2)=O)cc2c(nn1)CCC2 N1(C(c2ccc(C)cc2Br)=O)CC(NC(C2CC(O)C2)=O)CC2(CCC2)C1 C12(C(=O)OCC(c3ccco3)OCC)CC3CC1C2C3=O Cc1cc(=NCC#CCCO)[nH]cc1S(=O)(=O)N1CCC(C2COCCO2)CC1 c1(C(N(CC#C)C2CC2)=O)n[nH]c2c1CN(C(=O)C(CC)C(F)(F)F)C2 C=C(C)C(C)(O)C(=O)NC1CCC(CN(C)C(c2cc(OC)ccc2C)=O)CC1 CC(C)(C(=O)NCC1CN(C(C2CC2(Cl)Cl)=O)C1)C(F)c1ccccc1 C1(NC)CCCCN(C(c2cc(-c3ccccc3OC)no2)=O)C1 [N-]=[N+]=NCC(F)CCNC(C1CCCC(NC(=O)CN2CC=CC2)CC1)=O C1(NC(C(C)NC(=O)OC)=O)CC2CCC1C(NC(=O)C(F)(F)CO)C2 C1(C)(C(N(C(C)C)CCNC(C2C(C)C2C)=O)=O)CC2(CCC2)C1 N1(C(C(C)NC(C2CN(C(=O)Nc3ccoc3)C2)=O)=O)CCCC(F)CC1 Cc1ncc2n1CCN(C(=O)C(C)C(C)NC(=O)C(C)c1ccco1)C2 CC(C)(CNC(C1CCOC(=O)CC1)=O)CC(=O)NCC1CC(O)C1 C12(C(c3ccccc3)C3CC3)CCCC1NCC2.CCCC=CCCN c1(C(N2CCC(NC(CCCCCC#C)=O)C2)=O)cc2n(c1)CCS(=O)(=O)C2 N1(C(C2CC(=O)N(C3CCCCC3)C2)=O)CC2(C1)CN(C(=O)C1=CCCCO1)C2 c1(C(N2CCCC(N(C(C3CN(C)CCO3)=O)CC)C2)=O)ccc2c[nH]nc2n1 C(=O)(N=c1[nH]oc2cc(Cl)ccc12)Nc1c(C)nc(-c2ccn3nccc3c2)cc1 C(c1ccc(F)cc1)=CC(=O)NC1CC2(C1)CC2NC(=O)Cc1cccs1 c12ocnc1C(=O)NOC2.CC(C)(C)CC1CCN1C(=O)C(=O)NC1CC1 C1(NC(CNC(CC)=O)=O)CCCCC12CCCN(C(c1ccc(=N)[nH]c1)=O)C2 CONS(=O)(=O)c1ccc(C(=O)NC2(CCNC(C3CC(F)C3)=O)CC2)cc1 C1(F)(C(=O)NC(CCOC)CNC(c2cc(C)cs2)=O)CS(=O)(=O)CC12CCC2 N1(C(c2ccc(CC)cc2)=O)CC(CO)C2(C1)CN(C(c1nccn1CC)=O)C2 C1(C)(C(N2CCC(C(C)C(=O)NCCC3CC(O)C3)C2)=O)CCOCC1 c1(C(=O)NC(CNC(CCCC(=C)C)=O)CO)cc(N)c(C)cc1C N1(C(CNC(N)=O)=O)CCN(C(c2c[nH]cc2Br)=O)CC1 C1(C(=O)NC(c2cn(CC)nc2)C)CN(C(=O)C(O)C(F)(F)F)CCN1C Cc1nc(S(=O)(=O)N2CCCCC2C(N2CSCC2C)=O)cn1C c1(C(=O)NCc2c(C)nc(C)s2)n[nH]c2c1CN(C(=O)Cc1ccco1)C2 c1(CC(=O)NC(C2CCN(C(c3cc(O)cs3)=O)C2)C)ccc2[nH]ccc2c1 C(C(C(C)C(C)C)NC(c1nc(O)c(C)s1)=O)NC(CN(CCCCCC)C)=O c1(CNC(C2(CC)CN(C(C3(OCC)CCC3)=O)C2)=O)nnc(O)n1C C1(N(C(c2coc(CO)c2)=O)CC)CCCN(C(=O)CCOCC(F)(F)F)C1 c1(CC)nccnc1CNC(=O)C(c1ccccc1)NC(C12CSCC1C2)=O c1(CCC)nnc(S)n1CC(=O)NC(c1cn(-c2cncc(Br)c2)nn1)C N(C(=NCC1CC1)NCC(C(C)(C)C)OC)CC1(C(=O)OC)CCOC1 C1(N(C)C(c2cccc(CO)n2)=O)CCCN(C(=O)C(C)(C)C2CCCCO2)C1 C1(CC(=O)NCCF)CC(N=c2ccnc(C(F)(F)F)[nH]2)C1 N1(C(c2ccc(C(C)=O)o2)=O)CCC2(CCC(NC(=O)C(O)CC(N)=O)CC2)C1 C(C(=O)NCCCCNC(c1cc(C(C)(C)C)c[nH]1)=O)(C(C)C)OCC n1(C(C(=O)NCCC(C)NC(=O)CC2(N3CCCC3)CC2)C)cc(Cl)cn1 Cc1cc(C(=O)N(CCNC(=O)C(O)C2CCC2)Cc2ccccc2)cnc1F c1(C(=O)NCCNC(C2CC3(ON=C(C)C3)C2)=O)[nH]c2ccccc2c1Cl C(=O)(C(C)CC)NCC(=O)NCCC1CC(C(=O)NCC(C=C)O)C1 C(=O)(CC(C(C)CC)NC(C1CC(C)(C)CO1)=O)N(CCOCC)C N1(C(C2(CNC(CNC(CC)=O)=O)CCCO2)=O)CC(C2CC2)(COC)C1 N1(C(=O)NC(COC)C)CCC(NCc2cccc(CO)c2)CC1 C12(C(N3CCN(C(C4C(C)=CCS4)=O)CC3)=O)CCC(C1)OC2C C1(C(N2CC(C(CC)C)C2)=O)C2CCC(C2)N1C(C1(CC)CCCO1)=O c1(CC(=O)NCC2CCCCN2C(c2ccc(F)c(O)c2)=O)ccnc(F)c1F C=CCCCCCC(=O)N1CC(C)(NC(=O)CN(C)S(N)(=O)=O)C1 Cc1ccc2c(c1)OC(C)CN2C(C(=O)NC1CC(F)(F)C1)C1CC1(Br)Br C1(CC)(NC(N)=O)CCCN(C(C2CC23CC(OC(C)(C)C)C3)=O)C1 N1(C(C(C)C2CCOC2)=O)CC(C2CCN(C(=O)CS(=O)(=O)CCO)CC2)C1 C(CC(=O)N(C1CC1)CC1(O)CCC1)(C(C)CC)NC(c1ccc(C#C)o1)=O N1(CC(=O)NCCSc2cccc(Br)c2)CCC(C2CCNC2)CC1 N1(C(CN2CCN(C(C3C(CCC)C3)=O)CC2)=O)CCC(F)(C#N)C1 CC(C)(CC(F)C(=O)NCCc1nc[nH]n1)NC(C1CC12CC2)=O N1(C(c2c(SC)ccs2)=O)CCC(C)CC1CNC(=O)Cc1cc(C(C)C)no1 N1(C(C2(NC(CCCOC(C)(C)C)=O)CSC2)=O)CCCCC(F)(F)C1 C#Cc1ccc(CC(N2CCC(C(C)NC(=O)C(C)C(F)(F)F)CC2)=O)c(F)c1 C(=O)(C1=CCN(C(=O)C(C)C(F)(F)F)CC1)NC(CC)(C)C C1(CNC(=O)CSCC2CCCO2)CC2(CCN(C(=O)CSC(F)F)C2)CO1 c1(C(N2CC(CNC(C(C)(C)CF)=O)OCC2)=O)n[nH]c2nccc(Cl)c12 N1(C(C(C)(C)OC)=O)CC2CCCC(NC(=O)Cc3ccccn3)C2C1 N1(C(C)=O)CCCC2(CC(NC(=O)C(c3ccc(Br)cc3)(C)C)CO2)C1 N1(C(c2c(C)ccs2)=O)CC2CCC2(NC(c2ccc(C#N)[nH]2)=O)C1 C#CCC(CC(=O)OC)N(CC=C(Cl)Cl)CC1(C)CCCC(=O)N1 c1(CCC)c(NC(C2CSCCN2C(=O)C(O)CCC)=O)cnn1C S(=O)(=O)(c1ccc(F)c(SC)c1)N1c2c(ccc(SC)c2)CC1 CCC(C)C(O)C(=O)NCC(C1(O)CN(C(c2cnn(C)n2)=O)C1)(C)C c1(C(=O)NCC23N(C(C#CC(C)C)=O)CCC2CC3)ccc2c(c1)NC(=O)C2 N1(C(C(N2C(C)C(c3ccccc3)CC2)=O)=O)CC2C3CCC(C3)C2C1 c1(C2(C(N3C(CNC(C(C4COC(C)(C)O4)O)=O)CC3)=O)CC2)c(F)cccc1Cl Cc1cc(S(N)(=O)=O)oc1C(=O)NC1CCN(C(=O)CCc2nc[nH]n2)C12CC2 c1(C(=O)OC)ccc(=NCC2CC(NC(=O)CC(C)c3ccncc3)C2)[nH]c1C C1(NC(=O)CCF)CC(F)CN(C(C2CCN(Cc3ccccc3)C2=O)=O)C1 C1(NC(C(C(=O)OC)(C)F)=O)CN(C(=O)C(F)=C(C)C2CC2)C2(CCCC2)C1 C1(C(=O)NC2CCC(N(C(=O)CSC(F)F)C)CC2)C(C2CC2)C1(F)F C1(C(=O)Nc2nc(C)sc2)C(C2CC2)CCN1C(=O)C(c1ccn(C)n1)C C1(C(=O)NCC(C(C)C)(C)NC(C2CCC(C)(C)C2)=O)CC(C)(C)C(C)(C)C1 N1(C(c2cnco2)=O)CCN(C(C2(c3ccccc3)CCCCO2)=O)CC1 C=CC1(CC(=O)NOC(C)C)CN(C(=O)CCOCCOC)C1 C=C(C)CN=C(NCc1ccc(OC(F)(F)F)cc1)NCC1CCOCC1C C(c1ccnn1C)=CC(=O)N(C1CCN(C(c2cccnc2S)=O)C1)C Cc1cc(C(=O)N(CC(CO)(CO)NC(=O)Cn2nnc(C3CC3)n2)C)ncn1 Cc1ccc(C=CC(=O)NCCC2CN(C(c3[nH]c(C4CC4)nc3C)=O)C2)cn1 c1(OC)c(F)ccc2c(C(=O)NCc3ccc(Cn4cccn4)cc3)coc12 c1(C(N2C(CC)CN(C)C(=O)C2)C(=O)NC(C)(C)C)cc(C)nc2ccccc12 N1(C(C(C)S(N)(=O)=O)=O)CCN(C(c2csc(-c3cnccn3)n2)=O)CC(O)C1 N1(C(CC2(OC)CCCC2)=O)CCC(C)(NC(=O)CNS(=O)(=O)N(C)C)CC1 CCC(C)C(=O)NCC(=O)N(C)CC1(CNC(C2CCCSC2)=O)CC1 C1(F)(C(=O)NC(CC=C)CNC(C2CCCN(C(=O)NC)C2)=O)CCCCCC1 C(C1=NOC2CN(C(=O)CC(C3CC3)C3CC3)CC12)NC(c1nc(C)sc1C)=O C1(C(N(CCCOC)C)=O)CC(NC(c2ccsc2OC)=O)C(O)C1 C(CCCC(=O)NC1CCCN1C1CC1)N(C)C(C1CN(C(C)N(C)C)CCO1)=O c1(OC)ccc2c(c1)OCCC2C(=O)NC1CCC1CNC(c1ccsc1C)=O Nc1nonc1C(=O)NCCC1(C(=O)NC2CCCC2O)CC1 C1(OC)CC(CNC(=O)CCCCn2ccnn2)N(C(=O)CN2CCCS2(=O)=O)C1 c1(CC)nn(C)c(Cl)c1C(=O)N(CCCNC(C1CC(F)CN1C)=O)C C(=O)(CC(C)(C)c1ccc(F)cc1)NC(CNC(c1c(C)noc1)=O)C1CCC1 CCCCC(O)C(=O)N1CC(C(C)NC(C2CCNC2=O)=O)C1 C1(C(=O)NCC(N2C(C(=O)OC)CCCC2)=O)CC2CCC1CC2O C(=O)(C1=CSCCO1)NCC1CCC(NC(CN2CC(=O)NC2=O)=O)C1 C1(C(=O)NCc2ncc(C)[nH]2)CCC(N=[N+]=[N-])C1 N1(C(COC)=O)CCCC(C(C)(C)C(=O)N2CC(C)(OC)C2)C1 c1(C(N(CCN(C(C23CCOC(C)(C2)C3)=O)CC)CC)=O)n[nH]c2ccc(F)cc12 c1(OC)cnnc(OC)c1C(=O)NC(C)CNC(c1cn(C)cn1)=O c1(OC)cnc(F)c(C(=O)NC2CCN(C(=O)Cc3cncc(O)c3)CC2O)c1 C(=O)(C(F)(CNC(=O)CC1CC2C=CC1C2)C(C)C)NC(c1nn[nH]n1)CC c1(C(C)NC(C(C2CCCC2)NC(C(C)=CC=C)=O)=O)snnc1C C=CC1COCCN1C(=O)CC1N(C(=O)CC2CNC(=O)O2)CCC1(C)C c1(C(N(C2CCCN(C(C(CCC)O)=O)CC2)CC)=O)cccc([N+](=O)[O-])c1C c1(C(N2CC(NC(Cc3cccc(CC)c3)=O)C2)=O)ccc(Cl)c(C)c1Cl S(=O)(=O)(c1c[nH]c(=NCCC2CC(O)C2)cc1C)NCCC(C=C)(C)C c1(C(=O)NC2(C)CN(C(c3cnn(CC)n3)=O)C2)ccncc1C c1(C(N2CCC(NC(c3ncn(CC)c3)=O)C2C)=O)ccn2nccc2n1 Cc1ccc(C2CC2)c(C(N2CCN(C(=O)C3=CSCS3)CC2)=O)c1 C1(C(N2CCC(N(C)C)C2)=O)CC(O)CCN1C(c1ccc(Br)cc1O)=O c1(C(=O)NC(C(C)C)CCNC(=O)C2=CCCC2)ccc(S(=O)(=O)CCO)cc1 C1(N(C(=O)CC2CC2(Cl)Cl)C)CN(C(C2C3CC4C(C3)C24)=O)CC12CC2 N1(CCCC=C)CCC(C(=O)Nc2cnccc2C(F)(F)F)CC1 C(=O)(C1=NN(C)C(=O)CC1)NCC12OCC(CNC(c3cnc(C)o3)=O)(C1)C2 C12(CNC(C=C(CC)CC)=O)CCC(C1)N(C(c1ccc(C3CC3)cc1)=O)C2 C1(C(=O)NCC=CCNC(C(CC2CCCC2)N(C)C)=O)CC(C2CCCC2)C1 CC1=C(C(=O)NC2CCOCC2C(=O)Nc2cc(C)ccc2C)CCO1 c1(NC(c2cccc(CNC(c3c(C)nc(C)o3)=O)n2)=O)cc(O)ccc1C C1(C(=O)NCC2CN(C(CC3N(CC)CCOC3)=O)C2)Cc2ccccc2CO1 C1(NC(C(C)NS(C)(=O)=O)=O)CCC(CNC(c2cn(C3CC3)nn2)=O)C1 CC1(F)COCCN(C(C2(NC(C3CCC(=O)O3)=O)CCCCC2)=O)C1 C1(C(=O)NCCC2(OC)CN(C(COCCCCC)=O)C2)CC(C2CCC2)C1 Cc1ccc2sc(C(=O)N(CC(O)CNC(=O)CCOC3CC3)C)c(C)c2c1 c1(C(N2CC(NC(CC(=O)OC)=O)CC23CCC3)=O)cccc2c1ncn2C C1(C(N(CC(CC)NC(=O)C(C)(F)F)CC)=O)COC2(C1)CS(=O)(=O)C2 C(=O)(CCS(N)(=O)=O)NC(C1N(C(CCCCC)=O)CCC1)C C=CCC(CC=C)C(=O)NC(CC1CC1)C(=O)NOCCF N1(C(C2(C(C)NC(=O)CC3CCCC3C)CC2)=O)CCc2c(O)cccc2C1 N1(C(c2n(C)c(S)nn2)=O)CCCCC(NC(=O)CC(c2cccc(F)c2)O)C1 CCC(C(=O)N1CCOCC1)NC(=O)C(n1cc(Br)cn1)C O=C(CC1C2CCCC2N1C(c1c[nH]c(=S)cn1)=O)N=c1ccn(CCCO)[nH]1 C1(C(=O)NCCC(CNC(C(CC#C)C)=O)=C)CC2(C1)CS(=O)(=O)C2 C1(OC)CCC2(C(=O)NCC(C)NC(=O)Cn3cccn3)CC12 C(=O)(C1=CCC(F)(F)CC1)N1C(C(=O)NCCCNCC)CCC1 CC1CN(C(c2nc(Cl)ncc2Cl)=O)CCN1N1CCN(C=O)CC1.C1CC1 C(=O)(C(C)(COCCN(C)C)CC)N1CCC(N(C)CC)C1 C12(C(=O)NC3CCN(C(c4cc(-c5ccc(C)o5)[nH]n4)=O)C3)CCC(CO1)C2 C(c1cc(F)c(O)c(F)c1)=CC(N1CCCC(NC(C2(CC=C)CC2)=O)CC1)=O c1(C(N2CCC3(C(CNC(c4cc[nH]n4)=O)C3)CC2)=O)ccc2c(c1)OCCO2 c1(C(=O)NC2CCC(NC(c3cccc(SC)c3)=O)CC2)cc(F)cc(Cl)c1O N1(C(C(C)n2ccnn2)=O)CCC2(CCCC2NC(C2C=CCC2)=O)CC1 O=C(C1CCc2cc(F)ccc21)NC1CN(C(=O)Cc2ccsc2Cl)C1 CCC(C)CC(=O)NC(C)CNC(c1cn(C2CCOC2)cn1)=O c1(C(=O)NC(C)CN(C)C(C2CCOC2c2ccccc2)=O)ccc(N)c(O)c1 c1(CNC(C(CNC(c2cn(CC)nc2)=O)OC)=O)cc(C)cc(C)c1 CCC(C)C(=O)C(=O)NC1(C(=O)NCCCF)CCSC1 c1(C(C(=O)NCC(C)CN(C)C(C2(O)CC2)=O)O)cc(F)c(F)cc1F CCCC(C)(C)CC(=O)NC1CCN(C(=O)C(SCC)SC)C1.C1(N)CCCCC1 Cc1nc(Cl)ccc1CC(=O)NCC1CC1NC(=O)CC1(C#N)CCCCC1 c1(C(N2CCC(C(C)NC(=O)C#CC(=O)N(C)C)C2)=O)cnn2c1OCCC2 CC1CCN2N=C(C(=O)NCC3(F)CC(CNC(C4(Cl)CC4)=O)C3)NC2=N1 c1(OC)ccc(F)c(C(N2CCCC2Cn2cc(CC3(O)CCSC3)nn2)=O)n1 Cc1ccc(O)c(C(=O)N(C)CC=CC(=O)NCCCc2ncc[nH]2)c1 N1(C(C(CC)NC(C)=O)=O)CC2(C1)CN(C(C1(CF)CC3(CCC3)C1)=O)C2 c1(C(=O)NCC(=O)NC(C(C)C)C(C)NC(C2CN(C)C2)=O)ccc(Cl)cc1Cl c1(NC(=O)NC)ccc(Br)cc1NC(=O)NCC(c1cccc(Cl)c1)OC N1(C(C(C(C)C)C2CCC2)=O)CC2COCC2(C(=O)N(CC(C)(O)C2CC2)C)C1 C(=O)(CS(=O)(=O)N(C)C)N(CCC)CCNC(c1snnc1CC)=O c1(C(=O)NCCCC(C)NC(C(C)NC(=O)OC)=O)c(Br)n[nH]c1C C(C)(C)(CCCN=c1ccc(C#N)n[nH]1)NC(C1CCc2n(C)cnc2C1)=O Cc1n[nH]cc1CC(=O)N(CCCCCNC(=O)CSC(F)F)C C(=O)(C1=NOC(C)C1C)NCC1(O)CCN(C(Cc2cc(C)c(F)cc2)=O)C1 C1(CNC(c2c(C)ncs2)=O)CN(C(c2cn(CCN(C)C)nn2)=O)CC1O c1(OC)ccc(F)cc1CC(=O)NC1CCN(C(=O)C(Br)=C(C)C)CC1O Cc1cc(OC(c2nc(-c3ccsc3)nn2CCCO)C)ccc1F c1(OC(C(=O)O)CNc2nc(Br)ccc2Br)ccc(Cl)cc1Cl N1(C(CCCCSCCCC)=O)CCC(N(C(=O)Cc2nnc(C)o2)C)C(C)C1 N1(C(c2c(C)cc[nH]2)=O)CCCN(C(c2ocnc2C2CC2)=O)CC1C(C)C c1(C(=O)OC)cc(C)c(C)cc1C1=CCNCC1 C(=O)(C1=Cc2ccccc2OC1)NCC1CN(C(C(CCC(C)C)=O)=O)C1 CP(C)(=O)c1ccc(C(N2CC(NC(=O)C3=NOC(C4(O)COC4)C3)C2)=O)s1 C(=O)(CC1CC(C(C)C)c2ccccc21)NCC#Cc1cccc(OC)c1 Cc1cn2cccc(C(N3CCCC3CCCNC(c3ccoc3)=O)=O)c2n1 c1(C(=O)NC2CC(C)(CNC(CCCC)=O)C2)ccc(Br)c2cccnc12 C1(NC(C(C)CO)=O)CN(C(=O)CN(C)CCc2ccccc2)CC1O N1(C(c2nnc(C)s2)=O)CCC2(CCCCC2NC(=O)CN2CCNC(=O)C2)C1 c1(C(=O)NC(C)CCNC(c2cnc(Cl)s2)=O)cn2cccnc2n1 C(=O)(C(O)C(C)CC)N1CC(C(N)=O)(CNC(c2c(C)nc(CSC)s2)=O)C1 C(=O)(C#CC1CCCOC1)NC1CCN(C(C=Cc2ccc(OC)c(Cl)c2)=O)C1 CC1CN(C(=O)CN2CCC(C)C2)CCCN1C(c1ccn2ccnc2c1)=O c1(C(N(CCN(C)CC)C)=O)cc(C)cs1.C(=O)(C(C1CCCC1)OC)NC C1(C(N2C(C)(C(=O)OC)C=CC2)=O)CN(C(C23CCN(CC2)CC3)=O)CCC1(C)C c1(OC)cc(CN2CCCC(C)(CN(C)C)C2)ccc1OC1CC1.C1(=O)CN1 c1(C(N2CC(NC(C3CC(=O)NC3)=O)C(F)CC2)=O)cccc([N+](=O)[O-])c1Br C1(NC(c2c(C)oc([N+](=O)[O-])c2)=O)CC2CCC1CN(C(=O)C(C)(C)C(F)F)C2 N1(C(Cc2n(C)cnc2)=O)CCC(CO)(Cc2ccc(OC(F)(F)F)cc2)CC1 C#Cc1cncc(C(N2CCC(C(=O)NCC(C3CCC3)OC)(CC)C2)=O)c1 C(=O)(C1=NN(CC)C(=O)CC1)NC1CC(CCNC(Cn2ncc(CC)c2)=O)C1 N1(C(C(CCC)NC(=O)CCCC(C)C)=O)CCOCC(C)(O)C1 C1(CNC(C2(O)CC(C)(C)C2)=O)(CO)CCN(C(C2CCCCC2)=O)CC1 c1(N2C(C(=O)OC(C)(C)C)CCC2)ncc2cn[nH]c2n1 C1(NC(c2c(CC)cno2)=O)CCCCC12CCN(C(=O)C#CC1CCCC1)C2 N1(C(c2ccnc(Cl)c2)=O)CCOC2(C1)CN(Cc1ccc(F)c(Br)c1F)C2 C1(N(C(=O)C(F)n2cccn2)C)CCN(C(C2CC3(CCC3)C2)=O)CC1 C1(C(=O)NCCC(O)C2CC2)CN(C(=O)CC2COCCOC2)C2(CCC2)C1 N1(C(C(COC)OC)=O)CCC(C2CC2)(CNC(=O)Cn2ncc(C)cc2=O)C1 c1(C(N2CC3C(CNC(C(CC)=CC)=O)(C3)C2)=O)ccc2c(n1)CCC(C)C2 C(=O)(C(O)CC(F)(F)F)N(CCNC(C1(CCOC)CCC1)=O)C1CC1 Cc1cnc(CNC(=O)C(Cn2ccnn2)NC(C2CN3CCC2C3)=O)cn1 c1(C(C)C)cccc(C(N2CC(O)(C(C)NC(=O)C(C3CCOCC3)F)C2)=O)c1 N1(C(C(COC)(C)O)=O)CCC2(CCN(C(=O)C(C)C(C)C)C2)C1 C1(CC)C(C(=O)NCC2(C)CCOCC2)CCN1C(=O)C(CN(C)C)N(C)C CC1(C)OC2(C(=O)NCC3CCCN3C(=O)CNC(c3ccco3)=O)CCC1C2 C1(NC(c2c(CC)c[nH]c2)=O)CN(C(c2ccc(C(N)=O)[nH]2)=O)CC2(CC2)C1 c1(C(N(CC(C)NC(c2cc(C)nc(C)c2)=O)C)=O)cc(Cl)cc2ccncc12 C#Cc1cn(C)nc1C(N1CCC(N(C(C2(N(C)C)CCCOC2)=O)CC)C1)=O N1(C(c2occ(C)c2)=O)CC(NC(=O)Cc2csc(C(C)(C)C)n2)C(C2CC2)C1 C#Cc1ccc(CC(=O)NC(C)C(C(C)C)NC(=O)CN(S(C)(=O)=O)C)cc1 N1(C(c2cc(CNC(C(n3ccc(C)n3)C)=O)on2)=O)CC(O)CC1(C)C c1(CNC(C(C)C)=O)nnc2n1CCN(C(=O)CC1CC3CC3C1)C2 c1(OC)ccc2c(C(=O)NC3CN(C(c4cccc5oncc45)=O)C3)cnn2c1 C(=O)(C1=CCC(C)CC1)NCCOCCC(=O)NC(C=C)COC C1(O)(CNC(c2cn(C)nc2-c2ccccc2)=O)CCc2ccccc2C1 C(CN=c1[nH]c2c(c(=NC(CC3CCC3)c3ccccc3)[nH]1)CSC2)NC(C)=O C1(OC)CN(C(C2(C)CNC(=O)N2)=O)CC1C(=O)NCCC1CC1C C12(CNC(C=CSC)=O)CC(NC(C3CCCCC3C)=O)(C1)C1(CCOCC1)O2 C(=O)(CCCCC(=O)N1CC2CC(NC(c3coc(C)n3)=O)C2C1)NC c1(C(=O)NCC2CCCCN2C(C2CC23CCC3)=O)occ2c1CCCC2 C(=O)(C1=CC2(CCN(C(C3CC3(F)Cl)=O)C2)C1)NC1C(CN(C)C)C1 N#CC1CN(C(=O)Nc2cc(C(F)(F)F)ccn2)CCO1 c1(C(=O)NC2(CNC(C3C(COC)C3)=O)CCC2)cnccc1Br N1(C(=O)Nc2cc(CCCCC)cc(Br)c2)CC2CCCCC12C c1(NCCNC(=O)NCCOCCOCC)cccc(Cl)n1 C1(CC(=O)NCC2CC(C)(O)C2)(OC)CN(C(=O)CCc2ccccc2)C1 Cc1cc(O)ccc1CC(=O)N(C1CCCN(C(=O)CCc2cscn2)C1)C C1(C#N)(OC)CC(C(=O)NCCCC(C)NC(=O)CC2CCCOC2)C1 C#CCC(O)C(=O)N1CC(OCC(=O)N(c2cnccc2C)C)C1 c1(CCNC2(C)CC(C(F)F)C2)nc2ccccc2s1 Cc1cc(C(=O)N(C2CC(NC(=O)C(C)c3ccsc3)C2)C)cc(N)c1 c1(CC(=O)NCCCC(C)NC(C2COC(=O)N2C)=O)ccc(F)cc1 N1(C(CCOCC)=O)CC(NC(c2ccc3ncncc3c2)=O)CC12CCOC2 c1(C(=O)NC(C(C)NC(Cc2cc(C(C)C)no2)=O)C)ccnc(O)c1 CCC(CC(=O)N1CCCC1CNC(c1cc(N)cc(C)c1F)=O)CC(F)(F)F c1(C(=O)NC(CN(C(=O)CCOC)CC)C)ccc(CC(C)(C)C)cc1 c1(C(=O)NCCCCN(CC)CC)cccn2c(C3=CCC(C#N)CC3)cnc12 N1(C(=O)C(F)n2ccnc2)CC2CC(C(=O)NCCC3CC(F)(F)C3)(C2)C1 CC(CC(=O)NC(CCOCCO)C(N1CCCC(C)CC1)=O)C(F)(F)F Cc1ccc(=N)[nH]c1C(N1CCC(C)(NC(c2ccc(SC3CC3)cc2)=O)C1)=O n1(CC)cc(C(N2CCCC2CCC(=O)N2CC(OC(C)C)C2)=O)c(C)n1 c1(C(N(C2CCN(C(C3CC3C(C)(F)F)=O)C2)C)=O)cn(CCCF)nn1 c1(CCC)c[nH]c2ccc(NCC34CCCC3C4(F)F)cc12 N1(C(CCCN2CCN(C(C)C)CC2)=O)CC(NC(=O)OC(C)(C)C)CCC1C N1(C(CCCNC(C)=O)=O)CC2C(CNC(=O)C3=C(C)CC3)C2C1 c1(NC2(C(N)=O)CCN(S(C)(=O)=O)C2)nccn(C)c1=O n1(CC)nc(C(=O)N(CCCCC(=O)N(CCCCC(=O)NC)C)C)c(C)n1 c1(C(N2CCN(C(C)C)C(C)C2)C(=O)NC(C)C)ccc2c(c1)COC2 Cc1nc2ccccc2nc1C(=O)NC1C2CCN(C(=O)Cn3nccc3C)C12 N1(CC(=O)NCCC(C)CNC(C(CC=C)(C)CC)=O)CCc2ccccc2C1 CC(C)(O)C(F)(F)C(=O)NC1CC(O)CN(C(c2ccc(Cl)cc2)=O)C1 C12(C(=O)NCC3(COC)CCC3)CC(C)(CN1C(C1CCCS1)=O)C2 N1(C(CCSCC)=O)CCC(n2cc(CNC(=O)CCC#N)nn2)CC1 CC#CCC(C(=O)NCC(=O)NC)NC(c1ccc(C)cn1)=O c1(SCC(=O)NCC(CC)Oc2ccccc2F)ccc(-c2nn[nH]n2)cc1 C12(C(=O)NC3C(NC(CN(C)C)=O)C3)CCCCC(F)(C1)C2 C1(OCC(=O)N(CC(CN(C(c2nc(COC)sc2)=O)C)O)C)CCCC(C)C1 c1(C(N2C(C(N3CCN(CCCC)CC3)=O)C=CC2)=O)ncnc(C)c1C C1(C)(CNC(c2nc(CC)[nH]n2)=O)CCN(C(=O)C=CC2CCC2)C1 Cc1cncc(C(N2CCN(C(=O)Cc3ccn(C)n3)CC2CO)=O)c1C C=Cn1nccc1C(=O)NC1(C(=O)NCC(C)(C)C(=O)OC)CCCC1C Cc1cc(O)c(F)cc1NC(=O)CC(C)CNC(c1cc(CO)[nH]n1)=O C=C(C)C1OCCC1C(=O)NCC1CC(C)N(C(c2ccc(F)cc2)=O)C1 n1(CC)ncc(C(=O)NCC(C)(CO)NC(=O)CNC(c2ccccc2)=O)c1Cl C1(NC(c2c(C=C)cnn2C)=O)CCN(C(=O)C(C)SC)C12CCC2 CCCC(C)(O)CC(=O)N1CCC(C)(C)C(C(=O)NC(C)(C)C(=O)NO)C1 n1(CC(=O)NCC2(F)CCN(C(C(C)N(C)C)=O)C2)ccc2ccccc2c1=O C1(C(=O)NC2C(C(N(C(CC)CO)C)=O)COCC2)CCC(O)CN1C c1(C(N(C2CCN(CC)C2)CCC)=O)cc(S(=O)(=O)N2CCC2)c[nH]1.C(CO)SC c1(C(N2C(CNC(=O)CC3CC3)CCC2)=O)cccc(C2CC(F)(F)C2)c1 N1(C(C(C)(C)Cl)=O)CCC(C2CCCN2Cc2cn(CCN(C)C)nn2)CC1 N1(C(C2CCC(CC)O2)=O)CCOC(CC(=O)NCc2oc(C)nc2C)C1 CC1CCN(C(=O)Cc2ccccc2F)C1C(=O)NCCc1nnc(O)o1 CCC(C)(C)C(O)C(=O)N1CC(CNC(c2nccn2C)=O)C2(CCC2)C1 C(CC(=O)N(C1CCCC1)C)(C(C)(C)C)NC(CCCNC(C)=O)=O c1(C(C(=O)NCC(=O)OC)(C)NC(=O)CC2CCOC2=O)ccc(C(C)C)cc1 C(CC(C)CCNC(c1csc(C(C)(C)C)n1)=O)NC(C1(CCC)CCC1)=O c1(C(N(C(CC2C(CNC(C(C)NC(=O)NC)=O)C2)=O)C)C)ccncn1 c1(C(=O)NCCN(C(CC)=O)C)ccc(OC)c(C(C)C)c1 c1(CC(=O)N(C(C)CCNC(C2CC2Br)=O)C)cc(O)nnc1O C1(NC(COCCC)=O)CCCCCC1NC(c1cnn(C2CCC2)c1C)=O c1(OC)cncc(C(=O)NC2CC(CCNC(=O)C(C)(C)C3=CCSC3)C2)c1C C1(CC(=O)NCC=CCNC(=O)C(=O)Nc2ccccc2)(COC)CCOCC1 c1(NC(C)CS(N)(=O)=O)ccc(S(=O)(=O)NC(Cc2nccs2)CO)cc1Br C(=O)(CCC(CF)CF)NC1CC(C(=O)NCc2n(C(C)(C)C)ncn2)C1 N1(C(CC=CC)=O)CCC2CCC(C1)N2C(=O)C(c1cccnc1)OC C12(C(=O)NCC(C(C)(C)O)(C)C)CCCC1CCN2C(=O)CCC1CC1(C)C c1(OC)ccc2[nH]c(=NCCN3CCC(O)C3)nc(N3CCCC(CO)C3)c2c1 C12(NC(c3cc(O)ccc3F)=O)CCOCC1CN(C(=O)CCn1cccn1)C2 Cc1ccc(C(=O)NCC(C)N(C)C(C2(NC(c3cccs3)=O)CC2)=O)c(O)c1 C1(C(N2CCC(CNC(C3(N4CCN(C)CC4)CC3)=O)C2)=O)CC2CCC(C1)S2 Cc1c(Br)ccc2[nH]c(C(=O)NC3CC34CC(NC(=O)CC(C)(C)O)C4)cc12 Cc1nn(C)c(C)c1OCCc1nc(-n2cc(CCCC#N)nn2)cs1 C1(OC(C)C(=O)NC(C)(C)CN(C)C(c2cc(C(N)=O)c[nH]2)=O)CCCCC1 Cc1cccc(C=CC(N2CC3(C2)CN(C(c2ccc(Cl)nc2N)=O)C3)=O)c1 c1(C2C(c3n(CCO)nc(-c4ccccn4)n3)C2)c(Cl)cccc1Cl Cc1cccc(CC(=O)NC(C)(CO)C(=O)NCC2=CCCCC2)c1 c1(CC(=O)NCCN(C2CCCC(C)C2)CCOC)cccc(OC(C)C)c1 C1(O)(C(C)NC(C2COCCO2)=O)CCN(C(=O)Cn2cccc2)CC1 CP(C)(=O)CN1CC(C(=O)NC2CCN(C(c3c[nH]c(=O)cn3)=O)CC2O)C1 c1(C2(Cc3ncc(CC)s3)CC2)nnc(N(C)CC)n1Cc1cccc(F)c1 C=CCC(C)(C)C(=O)N1CCC(C(C)NC(c2cn(-c3ncccn3)cn2)=O)C1 C=C(C)CC(C(=O)N1CCCOC(C)C1)NC(=O)C(N=[N+]=[N-])C(C)C C1(C(C(=O)NC2COC2)N(C2CC(C(=O)OC)C2)C)CC2C(C1)C2(F)F c1(CNC(C(C)C2CCCC2)=O)cn(C2CCN(C(=O)C(C)(C)O)C2)nn1 C1(C(=O)NCC(CC)NC(=O)CCCC(N)=O)CC2CCC(C1)S2(=O)=O C1(C(N(C2CC(C(=O)NC)C2)C)=O)CCC(CNC(=O)COC(C)=O)O1 C1(NC(C(C)=CC)=O)CN(C(=O)CCOc2cccc(F)c2)CC12CCOCC2 CCCCC(CC(=O)N1CC2CC(C)C2C1)NC(c1ccc(O)nc1C)=O c1(OC)ccc(F)c(C(=O)NCCC2(NC(C3CCCC(C#N)C3)=O)CCC2)n1 C1(N)C2CC3C(C2)C13.N1(C(N(CCCCC)C(C)C)=O)CC(F)CC1CCO n1(CC(=O)NCC=CCNC(c2nc(C(=O)OCC)sc2)=O)ncc(C#N)c1N N1(C(c2cc(C)c(F)cn2)=O)CCCN(C(C2CCCOC2C)=O)C(C(C)C)C1 C#CC1(C(N2CCOCC(CO)C2)=O)CCN(C(c2c[n+]([O-])c(C)cn2)=O)C1 S(=O)(=O)(c1ccc(NCC2CCCC(C)(C)O2)c2cnccc12)NC(C)CO N1(C(c2nc(C(C)OC)oc2)=O)Cc2nccn2CC(NC(C2(OC)CC2)=O)C1 N1(C(C2(S(N)(=O)=O)CC2)=O)CCC2(CC1)OCCC2NC(c1cncc(Cl)n1)=O C1(C(N2CCCC2CNC(C2(COC)CC(=C)C2)=O)=O)CCCS(=O)(=O)C1 C1(CNC(CCN(C)CC)=O)CCN(C(C2CCC(CC)O2)=O)C12CC2 c1(C(=O)NCC#CCNC(CNC(=O)NC)=O)[nH]c(-c2cccc(C)c2)nc1C C1(C(=O)NCC(CC=C)NC(C2(F)CCS(=O)(=O)C2)=O)Cc2ccccc2CO1 CC(C)(O)C(F)C(=O)NCCC1(O)CN(C(C2CCCOC2)=O)C1 N1(C(C23C(C)OC(CC2)C3)=O)CCCC(F)(CNC(C2CC3(CC3)CO2)=O)CC1 C1(CC)CN(C(c2cc(OC)cs2)=O)CCC1N=c1[nH]c(C(C)C)nc(Cl)c1C CC(C)C(C)C(C)CC(=O)N1CCCCC(NC(=O)C(C)(C)CN(C)C)C1 n1(CC)nc(C(=O)NCCCC2(NC(c3cc(C)cnc3C)=O)CC2)ccc1=O c1(N2C3CN(C(c4cc(C)sc4)=O)C(C3)C2)nc(Cl)nc2c1cnn2C N1(C(C2(NC(C(C)CC3CCCC3)=O)CCCC2)=O)CC(F)(C2CC2)C1 N1(c2[nH]c(=NCc3c(C)non3)[nH]c(=N)n2)CCOc2cccc(Cl)c2C1 c1(C(=O)NCC2COCCN(C(=O)CC3=CCCC3)C2)ccnc2c1CCO2 C1(C)(CC(=O)NC(CC2CN(C(CNC(=O)NC)=O)C2)C)CCCCC1C CCC(C)CC(=O)N1CCC(O)(CN(C(=O)COc2ccccc2)C)C1 N1(C(c2[nH]cc(C(C)=O)c2)=O)CC2(NC(=O)CCC(C)C)CCC1C2 Cc1ccc(C)c(C(N2CC(C(N3CCC(=O)C(C)C3)=O)C2)=O)c1O Cc1cccc(C(O)C(N2CCOC(CNC(=O)C=Cc3cncn3C)C2)=O)c1 c1(C(c2n(CCC)nnn2)NC2(COC)COC2)ccc(OCC(F)F)cc1 C1(NC(c2cc(-n3ccnc3)ccn2)=O)(CF)CCN(C(=O)CC2C=CCC2)C1 c1(C(=O)NC2CCC(NC(=O)CCC3CCCCO3)C2)ccc(Br)cc1F C1(F)(CNC(C(CC(C)C)O)=O)COCCN(C(=O)CCn2ccnc2)C1 C(=O)(C1c2c[nH]nc2CCC1C)NCC1(CN(C(C2(OC)CCC2)=O)C)CC1 CCCCS(=O)(=O)CC(=O)N1CC2CC(CNC(C3CCOC(=O)CC3)=O)C2C1 N1(c2nnc(C3C(C)(C)OCCO3)o2)CCCC(C)(C(F)(F)F)S1(=O)=O Cc1coc(C=CC(=O)NC(C)CCNC(c2nn(C(C)C)nc2Br)=O)n1 C(=O)(C(F)C(=O)N(CCCNC(c1nnn(C2CCOC2)c1C)=O)C)OCC Cc1ncc(C(=O)NCC2CC2NC(C2CCOCC23CCC3)=O)cc1C#N Cc1cc(C(N2CC=CC(C(=O)NC34CC=CC(C3)OC4)C2)=O)c(C)nn1 c1(C(N(C)CC2CCN(C(C3CC4CCC(C3)S4)=O)C2)=O)cccc2cncn12 c1(C(=O)NC(CN(C(C(CCC)CC)=O)CC)C)cc(OC)nc2ccccc12 N1(C(c2c(C)n(CCO)cc2)=O)CCCC(N(C)C(C2CCS(=O)(=O)C2)=O)CC1 N1(C(c2ccncc2O)=O)CC2CC1CN2C(C1C2CC3C(C2)C13)=O N(C1CCCc2cc(O)ccc21)c1ncc(C(=O)OC)cc1F c1(CC(=O)NCC(C2CC2)NC(=O)CNC(=O)C(F)(F)F)nnnn1CC(F)(F)F C(CCNC(C12CC1CCN2C(=O)CC1(C)CCC1)=O)(C(C)C)OC c1(OC)cncc(NC(c2ncccc2NCc2cnccc2Cl)=O)c1 C1(NC(C(C(=C)Cl)(C)C)=O)CC2CCC(C1)N2C(C1CCc2ncncc2C1)=O N1(C(C(C)n2cncn2)=O)CCC2C(CCCN2C(c2cnn3c2CCC3)=O)C1 n1(CCNC(C2(CCO)CC2c2ccc(Cl)s2)=O)cc(Cc2ccccc2)nn1 C1(NC(C(C=C)O)=O)CC(F)CN(C(=O)CCN2CCOCC2)C1 c1(C(C)=O)cccc(C(=O)NCc2ncc(C(=O)NC3CSC(C)C3)cn2)n1 Cc1ccc(C(=O)NCC2CCC(NC(=O)C3=COCCC3)C2)c(N)n1 C1(N(C)C(c2cc(C3CC3)cs2)=O)CCC(NC(=O)CC=CC(C)(C)C)CC1 c1(C(=O)NCC(CC(F)(F)F)NC(CC=C)=O)ccc2nc[nH]c2c1 n1(CC)nccc1C=CC(=O)NC(C)CC1CN(C(c2ncsc2C(C)C)=O)C1 C(=O)(CC(C)C(C)(C)N)NCC(N1CCC(CC)CC1)=O c1(OC)cc(CC(=O)OC(c2ccc(C(C)C)cc2)C)ccc1Br c1(NC)cc(Cl)ccc1C(=O)NCC1CC1NC(=O)CN1C(=O)CN(C)C1=O C(=O)(C(C)CCCC(C)C)N1CCC(CC(N2C(CO)CC(OC)C2)=O)C1 N(C1CC(C)n2ncnc21)C(c1nccc(CNC(c2c(C)c[nH]c2)=O)c1)=O C1(CCNC(c2ccon2)=O)CC(F)(F)CN1C(=O)COC1CCCOC1 C=CCCC(C(=O)N(C1CC2CCC1O2)C)NC(=O)C(O)CCCC C1(C(N(CCCCN(C(Cc2c(C)scc2)=O)C)C)=O)CC(=O)C12CCCC2 CCC(C)(C)C(=O)NCC(CC(C)C)NC(c1cccc(C2CCCC2)c1)=O CC1(CNC(c2csc(CO)n2)=O)CCN(C(=O)Cn2ccc(C3CC3)n2)C1 N1(C(c2snnc2C)C(=O)NC(CC)(C)C)CCOC(c2nccs2)C1 N1(C(C2C(CC)CCC2)=O)CC2CCC(NC(=O)CCc3cnn(C)n3)CC2C1 N1(C(c2ccc(Br)c(Cl)c2)C(=O)NCCCOC)CCN(C)CC1(C)C.CC N1(C(C)=O)CCCC1C(N1CC(C(C)NC(=O)C(F)(F)Nc2cnn(C)c2)C1)=O C(=O)(C(C)CC(=O)N1CCN(C(C2CCCC2)=O)C(c2cccc(F)c2)C1)OC CCC(CC(F)(F)F)C(=O)N1CCOC(CN(C)C(c2c[nH]cc(Cl)c2=O)=O)C1 CCCCC(F)(F)C(=O)NC(COC)CC(=O)NCC(=O)N(CC)OC N=c1cc[nH]cc1C(N1CCN(CCNC(c2cc(C3CCC3)on2)=O)CC1)=O c1(C(=O)NC2CN(Cc3c(C)cccn3)CC2F)cc(C)n(C)c1C C1(NC(c2ccc(SC(C)C)cc2)=O)CCN(C(c2cc(Br)n[nH]2)=O)CC1C c1(CC)ccc(OC)c(C(=O)N(CC(C)NC(=O)C(CC)C(=O)OC)C)c1 CC(C)C(F)(CNC(C1(CF)CCOCC1)=O)C(=O)N1CCOC(CC2CC2)C1 N1(C(C(CC)N(CC)CC)=O)CCN(C(c2ccc(C)c(N)c2)=O)CC(CO)C1 c1(N(CC(=O)NCC(CNC(CCOC)=O)CO)C)sc(O)nc1C N1(C(CC2(CCC#C)OCCO2)=O)CCN(C(=O)C(O)CCSC)C(CCO)C1 C(=O)(CC1CCOc2ccccc21)NCC(C)CNC(c1ccc(O)c(Cl)n1)=O C#Cc1cc(NC(=O)C=CCC(C)(C)NC(c2cnc(OC)nc2)=O)ccc1C c1(C(=O)NCCC(CNC(C2CCC(SCC)CC2)=O)O)c(F)cc(O)cc1F C(=O)(C#CC1CCCOC1)N1CCC(OCCNC(=O)Cc2ccc(Cl)cc2)C1 CCCCC(O)CC(=O)N1CC2CCC(C1)C2NC(=O)C(C)=C1CCCC1 N1(C(C2C(OCC)C2)=O)CC2(CCC2)CC1CNC(c1ccc(Cl)s1)=O C1(NC(=NCCC)NCC(c2cccc(Cl)c2)CO)CCC2(C1)OCCO2 c1(C(=O)NC(C2CCN(C(c3cccc(F)c3F)=O)C2)C)ccc(Cl)c(F)c1F Cc1ccc(C=CC(N2CC3C(C(=O)NC4CCCN(C(C)C)C4)C3C2)=O)s1 S(=O)(=O)(c1c[nH]ccc1=NC(C)COCCOC)N(CC=C)CCO N1(C(C)=O)CCOCC1CSC1CCN(C(=O)Cn2cc(C(C)O)nn2)CC1 c1(C(=O)NCCC2(NC(C3CCCSC3)=O)CC2)ccc2c(c1F)CCC2 C(C)(CC=C)(CC=C)NC(CONC(C1CC(C#C)(O)C1)=O)=O c1(C(N2CCC(O)(C(C)NC(CCCC=C)=O)C2)=O)nccn2cnnc12 C1(CC(=O)N(CC(O)CNC(c2csc(Cl)c2)=O)C)CCCC(C)(C)C1 c1(N(C(CNC(C2(C=C)CCC2)=O)C)C)nc(OC)c2ccccc2n1 C=CC(O)C(=O)N(CC(O)CNC(c1c[nH]nc1-c1ccn(C)n1)=O)C c1(C(=O)NCC2N(C(C(C(=C)C)(C)C)=O)CC2)cccc2[nH]c(-c3cccs3)nc12 C1(C(=O)NC(CC)CCOC)CCCCCN1C(=O)C(=O)C(C)C C1(C(=O)NCCN(CCC)C(C2CCSCC2)=O)CCCC(CC(F)(F)F)C1 Cc1cc(CCC(=O)NCC2(CO)CN(C(=O)CC3CCOC3C)C2)no1 c1(CC(C(=O)NCCC(C)NC(COCCSC)=O)O)ccc2ccccc2c1 N1(C(C2(COC)C=CCC2)=O)CC2CCC2(CCNC(C2(O)CCCCC2)=O)C1 CC1(C)CCc2[nH]nc(C(N3CCC(NC(C4CC(CCF)C4)=O)CC3)=O)c2C1 c1(C(=O)C(c2cn(C3CC(NCCS(=O)(=O)N(C)C)C3)nn2)=O)ccc(F)cc1 c1(C(N2CC(CC(=O)NC3CCCN(CC)C3)C(C)C2)=O)cc(C)cc(C#N)c1 c1(C(N2CCC(O)(CNC(C(C(C)C)(C)C)=O)C2)=O)cc(C#N)ccc1N c12cnc3c(c1C)N(CCO3)C(=O)C2.c1(OC)ncccc1-c1ncon1 CC1(C)C(NC(c2cnc(S)nc2)=O)CC1CC(=O)NCCC(F)(F)CO N1(C(C(=Cc2cnc[nH]2)C)=O)CC2(CCN2C(=O)C(CO)NC(=O)C(C)C)C1 C(C(COC)C(=O)N1CCC(CN(C)C(C2(CSC)CC(F)(F)C2)=O)C1)OC N1(C(C23CCC(OC)C2C3)=O)CC2(CCC2)CC1C(N1CC(=O)NC(=O)C1C)=O c1(C(N(C(CCNC(CCC(C)C)=O)C)C)=O)cccc2c1OCC2(C)C N1(C(C(C=C)(F)F)=O)CCc2[nH]nc(CNC(=O)C(O)CCC)c2C1 Cc1ccc(F)c(C(N2CC3C(CNC(=O)COCC(F)F)C3C2)=O)n1 C1(C(=O)NC2C(NC(=O)CC3OCCCOC3)CCC2)CC2CCC(C1)O2 n1(CC)ncc(C(=O)NCCOC2CN(C(c3sccc3C3CC3)=O)C2)c1Cl N1(Cc2ccc(-c3c(F)ccc(C(NOC)=O)c3)cn2)CCC2(C1)CC2(F)F C1(CC)C(NC(c2ccc(COC)cc2)=O)CCN1C(=O)C1=CCCS1 C1(C(=O)NC(C(=O)OC)C(C)C)CN(C(=O)CN2CCCCC2=O)CC1(C)C C1(C(=O)NCCC2CCCN(C(c3ccc(O)cn3)=O)C2)CC2(CCC2)CO1 C1(N(C(Cn2cnc(=N)[nH]2)=O)CCO)CCCN(C(C2CC2(F)F)=O)C1 C(=O)(C1=C(Cl)CC1)NC(C(=O)NCC1CC(O)(CN)C1)CC1CCC1 CC(O)C(C)CNC(C1CCCC1CNC(=O)CC(C)n1cccn1)=O c1(-c2c(C)csc2)nc(C(C)C)nn1Cc1cccc(F)c1 c1(C(=O)NCCCN(C(CNC(c2c(C)occ2)=O)=O)C)ccc([N+](=O)[O-])nc1 c1(CC(N2C(CC(=O)OCC)C(=O)NCC2)=O)ccc2c(cnn2C)c1 C1(NC(COCCC#C)=O)CCCN(C(c2cnn(C)c2C2CC2)=O)CC1F c1(CN2CCN(C(C(N3CC(C)C(N)C3)=O)=O)CC2)c[nH]c2cccc(Cl)c12 c1(OCC)ccc(C)nc1C(=O)NC1CN(C(=O)CNC=O)CC1(C)C c1(-n2cc(CCC3N(C(c4[nH]cc(C)c4C)=O)CCC3)nn2)cc(Cl)cnc1Cl C1(C(c2cccnc2)=O)CN(C(=O)CCCc2cn(C3CCC3)nn2)CCO1 c1(CS(C)(=O)=O)ccc(C(=O)NC2(CF)CCN(C(=O)CNS(N)(=O)=O)C2)cc1 c1(C(N2CCCC(N(C(C=CC=CC)=O)C)CC2)=O)ncnc2ccsc12 Cc1cnc(C(N2CCOC(CCNC(=O)C(C)CF)C2)=O)cc1Br C1(NC(CN(C2CCSC2)C)=O)CN(C(c2csnn2)=O)CC12CCOCC2 c1(NC(C2=C(C)CNC2)=O)ccc(N=c2cc[nH]cc2)cc1 C(N=c1[nH]c(Cl)nc2c1CCC2)C1CC(NC(=O)C(F)C(F)(F)F)C1 n1(CC)c(CNC(C2CN(C(=O)C3=CCSC3)CC2F)=O)nnc1O N1(C(c2ccc(NC(C)=O)cn2)=O)CCCC2(NC(C3CN(C)C3)=O)CC2C1 CCCCC(CNC(=O)C(C)COC)NC(=O)C(C)(C)C1CCOCC1 Cc1nsc(C(N2CC(C)C2C(=O)NCCC(O)C2CCC2)=O)c1N N1(CC)CCn2cc(-c3ccc(COC)cc3)nc2C1.c12cc(nc(C)n1)N2 N1(C(C(C)C2(O)CCC2)=O)C(CC(=O)NCC2(CCCO)CC2)C2CCCC12 Cc1coc(CNC(=O)C(C)NC(=O)C(C2CCCCC2)F)n1 C1(CNC(C=C(CC)CC)=O)CC(C(=O)N2CCC(OCC(C)C)C2)=NO1 N(C1CCc2ccc(F)cc21)S(c1c(C)n(-c2ccccc2)nc1)(=O)=O N1(C(Cn2nc(C)c(C)c2C)=O)CCN(C(=O)CSC(C)C)C(C)CC1C C(=O)(C1CCc2ccc(Br)cc21)NC1(C)CCN(C(C2CC=CC2)=O)C1 c1(CC)nn(C)cc1NC(=O)CC(C)NC(=O)CC1(O)CCOC1 C1(NC(c2cnc(C3CCCO3)s2)=O)CC2CC1CN(C(C1CC1CF)=O)C2 C1(CC)CCCN(C(=O)CCN(C(c2nccnc2C)=O)CC2CC2)C1 C1(C2C(N)C2)CCN(C(=O)C(CC2CCCC2)CN)CC1 C1(C(=O)NCC(CC(C)C)NC(=O)C(C)(C)C(C)C)CCOCC12CCC2 N1(C(c2n(CC)ncc2)=O)CC=CCC1C(N1CC2CC2(CC)C1)=O C(=O)(CCC(=O)C(C)(C)C)NC(C(N1CC(C)CC(OC)C1)=O)C(C)C C1(NC(C=C(COC)C)=O)CN(C(=O)CN(C)C)C2(CCCCCC2)C1 C1(C(=O)NCC2N(CC)CCC2)CN(C(c2cnn(C)c2N)=O)CC12CC2 c1(C(=O)NC(CC)(C)CNC(=O)C(F)=CCCF)cnc2n1CCCC2 C(CCCC(=O)Nc1cnn(C)c1C)OCC.C12(CCC1)N(C1CC1)C2=O C=C1CON(C(=O)C2CCCN(C(C3(F)CC3)=O)C2)C1 N(C1CCCc2ccoc21)C(c1cccc(NC(=O)OC)c1)=O Cc1cc(C(=O)NCC(C)N(C(=O)Cc2cncs2)C)c(Cl)cc1N O=C(CCCn1cc(CNC(=O)C2CC2)nn1)C1CC(=C2CC2)C1 c1(C(C(=O)NCCCC2CC2)N(CC=C)CC2CC2)cc(C)c(Br)cc1C C#CCC(CC(=O)NCC(C)N(C)C(=O)OC(C)(C)C)NC(=O)C(C)(O)CC#C c1(C(N2CC3CN(Cc4cscn4)CC3C2)=O)cn2cc(F)ccc2n1 c1(OC)ccc(CN2CCC(CC(N3CCN(C)CC3CO)=O)C2)c(Cl)c1OC Nc1cc(C(N2CCC3C(NC(c4cccc(Br)c4F)=O)C23)=O)cc(F)c1 N1(C(CC)CC)CC(C(=O)NC(C)C(C)(C)NC(=O)Cn2cnnn2)CC1=O N1(C(c2cc(C)no2)=O)CCC2(CCCN(C(=O)COCCF)C2)CC1 c1(C(N2CC(NC(CC3CCC(C)O3)=O)C2)=O)cccc(N)c1Br N1(C(c2cnc(C(N)=O)s2)=O)CCC2(CC1)CN(C(C1CC13CC3(F)F)=O)C2 C(=O)(C1=Cc2ccccc2C1)N1CCC2(C(C(=O)NCCOCCC#C)C2)CC1 N1(C(C(=O)NC(C)CCc2ccncc2)=O)CCc2cc(Br)ccc2C1C1CC1 n1(C(CC)C)nc(Cc2ccccc2)nc1-c1sc(Cn2cncn2)nc1C N1(C(C2(C(N)=O)CC2)=O)CC2CC1CC2NC(=O)CCc1cc(Br)cs1 c1(NCCCNS(CC)(=O)=O)nc[nH]c(=NCC(=O)NC2CC2)c1C N#Cc1ccc(CNC(=O)C(Cc2ccsc2)NC=O)nc1 c1(SC)ccc(Cl)c(CN2CCN(C(=O)C(N3CC(C)C(C)C3)=O)CC2)c1 C#Cc1ccnc(C(N2CCC3CC23C(N2CCC23CC(O)C3)=O)=O)c1 CC(C)CC(O)CC(=O)NCC1CC1CNC(c1cc(CC(C)C)on1)=O C1(NC(C(C=C)O)=O)COCCC1NC(c1cc(C)ccn1)=O.n12cc(nn1)C2 C1(NC(c2cnc(C)s2)=O)CCN(C(C2C3CC4C(C3)C24)=O)C(C)C1 C(=O)(C(F)C(F)(F)C(F)(F)F)N1CC(O)(C(C)(C)CNC(c2cnco2)=O)C1 c1(COC)cc(F)c(C(=O)NCC2C=CCN2C(=O)CO)c(F)c1 CCCCCC(C)CC(=O)NC(CCSC)C(=O)NCC(C)(F)CC N1(C(c2ccccc2Cl)=O)CCC2(C(N3CC([N+](=O)[O-])C3)=O)CCCC12 N1(C(C(C)=C2CC2)=O)CC(CNC(c2cc(O)cs2)=O)C(C)C1 c1(C(=O)NCC(Cc2ccccc2)NC(C)=O)ccc2c(O)nc(=O)n(C)c2n1 c1(SCC(N2CCCC(N(C(c3nc(C#C)sc3)=O)C)C2)=O)ccc(C)c(C)c1 C(CCC(C(=O)N1CCCC1CF)NC(=O)COC1(C)CCC1)OC c1(NC(N2CCC(NCCCc3c(OC)cccc3)C2)=O)nnc2n1CCS2 c1(CC(N2CC(NC(C3CC(C(F)(F)F)CO3)=O)C2)=O)cc(F)ccc1Cl C(c1ccccc1Cl)=CC(=O)NCCCCC1CN(C(C2(C)CCCO2)=O)C1 CCCCCCCCNC(C12CC(NC(=O)CCNC(=O)NC)(C1)C2)=O C12(CNC(=O)C=CC3CCC3)CCC(C1)N(C(c1ccccc1Br)=O)C2 C12CCC(C1)NC(=O)C2.c1(C(=O)N(CCO)C2CC2)ocnc1C(F)F c12csc(n1)NC(=O)C2.C(=O)(C(C)=C1CC1)N(CCOC)C(C)C CON=C(C(=O)N1CC(N(C)C(c2ncccn2)=O)C1)c1ccco1 c1(OC)nc(Br)ccc1C(N1CCCC1C(=O)Nc1ncccc1OC(F)F)=O C(CNC(=O)CCc1ccc(N)cn1)(C(C)(C)C)NC(CCc1n(C)cnc1)=O CC1(C)CCCC1CN=C(NC1CC1)NC1CCC(C)CC1 C(=O)(C(O)C(C)C)NC(CCNC(C1(SC)CC(O)C1)=O)C N1(C(C(C)OCC)=O)CCCC(NC(c2ccc(NS(=O)(=O)CC)cc2)=O)C1C C1(NC(c2c(NC)scn2)=O)CN(C(C2CCn3nnnc3C2)=O)CC(C)(C)C1 C(C(F)(F)C(=O)N1CCC1CNC(C1(C)C=CCCC1)=O)OC c1(OC)cncc(C(N2CC(CNC(=O)CC3COCC3O)C2)=O)n1 C1(C(N(CC(C)OCC)C)=O)CCN(C(=O)OC(C)(C)C)CC1[N+](=O)[O-] CCCCC(CC(=O)NC(C)Cc1cnccn1)NC(=O)CC1CCN(C)CC1 c1(C2CN(C(C3C(C)CCN3C(c3c[nH]c(=S)cn3)=O)=O)C2)ccc(F)c(F)c1 C1(CN(C(C(Br)=C(C)C)=O)C)CN(C(=O)CC2(O)CCCC2)CC12CC2 c1(C(=O)NC2CCN(C(C(CC)CCOC)=O)CC2F)cccc2cnccc12 C(=O)(CCCCN(C(=O)CNC(C)=O)C)N1CC(CC(C#C)C)C1 CC1(C)CCC(F)(F)CC1NC(c1cccc2c1CNC2)=O CC(CC(=O)NC1CC(CNC(=O)C(c2cccc(F)c2)F)C1)C(F)(F)F O=S(=O)(c1c[nH]ccc1=NC1CCSC2(CCC2)C1)NCc1cc(Cl)sc1Cl c1(OC)ccc(F)cc1CC(=O)NC(C)CCCCNc1nccc(OC)n1 c1(-c2scc(CN3CC(C(C)NC(c4nc(Cl)cs4)=O)C3)n2)ccccc1Cl C1(CNC(=O)C(O)CCNC(C2(O)CCSC2)=O)CC2CCCC2C1 C1(C(=O)NC2CC3CN(C(C(c4n(C)ccc4)=O)=O)CC32)CC2(C1)CC(C)(C)C2 c1(OC)c(F)cc(C(=O)NCC(C)NC(=O)C(F)(F)c2csc(C)c2)c(N)c1F c1(C(=O)NC2CCCC(NC(C3(N(C)C)CCC3)=O)C2)c(F)cc(F)cc1Cl C1(C(N2CCN(CC#CC)CC2)=O)CC(NC(=O)CCCC(N)=O)C12CCC2 c12cc(C)c(o1)C(=O)NC(C(C)C)C(C)NC(=O)CNC2=O.c1(C)cccs1.CC c1(C(=O)NC2CC(CNC(c3nccc(C)n3)=O)OCC2)ccc([N+](=O)[O-])s1 C(=O)(C(O)CC[S+](C)C)N1CCN(C2CCN(C(c3nccc(C)c3)=O)C2)CC1 c1(C(=O)NCCN(C(=O)CC2CCC(=O)N2C)CC)cc(S(N)(=O)=O)cnc1C c1(OC(C(=O)NCCN(C(=O)C(C)OC(=O)C(C)(C)C)CC)C)cccc(C)c1 CC1CCCC(NC(C2(CNC(C3CN(C)C3)=O)CCCO2)=O)C1 c1(C(=O)NCCC(C)N(C(=O)CSC(F)F)C)nc2cnccc2s1 N1(C(C(C)NS(CCCC)(=O)=O)=O)CC2CC1CN2C(C1CCC(=O)NC1)=O c1(C(=O)NCC2N(C(Cc3cccc(C)c3)=O)CCC2C)ccc2nnnn2c1 C1(C(N2C(CC)(CO)CCC2)=O)CC12CCN(C(=O)CCCC(C)=O)CC2 CCC(O)C(C)C(=O)NC1CCCC1NC(=O)CCOCc1ccccc1 Cc1cccnc1-c1cn(CC(c2ccccn2)N(C)C)nn1 c1(CC)cccc(C(N2CC(CNC(c3c(C(F)(F)F)coc3C)=O)C2)=O)c1N CC1(C(N2CC3CC2CN3C(C2(CO)CCC2)=O)=O)Cc2ccccc2C(=O)O1 Cc1cccc(C)c1CNC1CCNC1=O N1(C(C)=O)CCCC1C(=O)N(C1CCCC1)CCC1CN(c2nncs2)C1.C(=O)N C1(CNC(C(CC)=CC)=O)CC12CCN(C(C1CCn3ncnc3C1)=O)CC2 CN1C2CCCC1CC(OC(c1cn(-c3ncccn3)cn1)=O)C2 Cc1ccc(C(=O)NCC(C2CCN(C(C3CC(F)C3)=O)CC2)(C)C)nc1O Cc1cc(=O)n(C)cc1C(=O)NCC1(O)CCN(C(C2(C(F)F)CCCC2)=O)C1 c1(C(=O)NCCC2(C(=O)NCC(C(C)C)OC)CCC2)ccn(C)c(=O)c1 C(c1ccc(Cl)c([N+](=O)[O-])c1)=CC(=O)NCC(N(C(C(C=CC)O)=O)C)C1CC1 N1(C(C(CCOC)NC(=O)CC(O)C2CCCC2)=O)CCC(N=[N+]=[N-])CC1 C1(NC(CC(C)N(C)C)=O)CC(C)CN(C(c2ccc(C#N)s2)=O)C1 CC1(C)CC(O)(C(=O)NCC2CCCC2NC(=O)C(C)(C)c2ccns2)C1 C1(NC(C(C)n2cccn2)=O)C(C)(C)CN(C(c2ccncc2N)=O)CC1(C)C N1(C(Cc2c(SC)cccc2)=O)CCN(C(c2cc(OC)ccc2N)=O)C2CC12 c1(C(=O)NCC2CC(NC(c3c(CC)ocn3)=O)C2)cc(OC)ccc1C c1(C(=O)NCc2scc(C#N)c2)ccc2nc(-c3ccc4nsnc4c3)sc2c1 N1(C(COC2(C)CCC2)=O)CCCCCC1C(N1CCC1)=O C(=O)(C1=CCC(C)CC1)N1CCC(CC=C)(C(=O)NC(CO)C(C)(C)CO)C1 C=CCC(C)(C)CC(=O)N1CC2CCN(C(c3cc(OC)nc(Cl)c3)=O)CC12 c1(C(=O)NCC(CN(C(COC)=O)C)C)ccc(OCC(F)F)nc1 C(=O)(C1CCCc2ncccc21)N1CC(N(C)C(C2C=CC=CC=C2)=O)C(O)C1 c1(CC)cc(N)ccc1C(=O)NCC1CCN(C(C2CC3CC2CC3O)=O)C1 Cc1cccnc1CCN(C)Cc1csc(N(C)C(=O)OC(C)(C)C)n1 c1(-c2ncc(C(=O)NC(C)CN(C)C)nc2)ccc(S(=O)C(C)C)cc1 N1(C(c2cnc(C(C)C)nc2)=O)CCN(C(C2CNC(=O)C2)=O)C(CF)C1 Cc1ncc(NC(C2CC(F)CN(C(c3ccc(C4CC4)cc3)=O)C2)=O)cc1Cl c1(NC(c2ccc(CC)cc2)=O)ccc(NC(C2CC(C)(CC)C2)=O)cc1C c1(C(=O)NCC=CCNC(C(C)CC(F)(F)F)=O)c[nH]c2cccc([N+](=O)[O-])c12 C(=O)(C1SCCc2ccccc21)N(CCNC(c1nc(C#C)sc1)=O)C1CC1 C(C)(CCC(=O)N1CCOCC1CCNC(c1nccnc1N)=O)OCC Cc1ccc2nc(C(=O)NCC3CCN3C(=O)C#CC3CCCCC3)cn2c1 C(c1ccccc1C#N)=CC(=O)NCCCCC(C)NC(c1cn(C)c(O)n1)=O c1(C(=O)NC(CC=C)CNC(=O)CC(C)F)ccc(OCCF)cc1 Cc1ccc([N+](=O)[O-])c(C(N2CCC(C)(NC(c3ccoc3C3CC3)=O)C2)=O)c1 C1(CNC(C=CC2(NC(=O)CC3CCN(C)C3=O)C(C)C2)=O)CC2(CC2)C(=O)O1 Nc1cc(F)cc(F)c1C(=O)NCC(F)CNC(c1ccsc1C(F)F)=O N1(C(c2c(C#N)cccc2)=O)CCCc2cccc(O)c21 Cc1ccc(C(=O)NC23CC(C2)N(C(=O)CCn2cccn2)C3)c2c1NCCC2 O=C(C1=NN2CCCN=C2N1)NC1CCCC1NC(C1CCCC1C1CC1)=O c1(C(=O)NCC23C(CN(C(CCCC(=C)C)=O)C2)C3)cc(F)cc2nc(S)[nH]c12 N1(C(c2ccc(C)c(C)c2)=O)CCN(C(c2ocnc2C)=O)C2CCCCC12 Cc1c(C(=O)NC2CCC2NC(=O)Cc2cnc[nH]2)oc2ccccc2c1=O CC1CN(C(=O)CSC(F)(F)F)CCC1NC(C1CCC(C)(O)CC1)=O CCC(CN(C)C)CC(=O)N1CCCCC1CNC(C1(F)CCOC1C)=O c1(C(=O)NCC(F)CO)nsc2cc(-c3cnn(CCCO)c3)ccc12 N1(Cc2cc(C)nn2-c2ccccc2)CCC(C)(C(c2ccccc2)=O)CC1 C1(NC(c2ccn(C3CC3)n2)=O)C2CC3C(C2)C13C(=O)Nc1cc(C2CC2)on1 CCCC(CC(=O)N(C1CCCC1)CC)NC(=O)C(O)CC C1(NC(c2c(CC)n(-c3ccccc3)nn2)=O)CC2CC1N(C(=O)C(C)(Cl)Cl)C2 C1(CNC(CCCC#C)=O)CN(C(=O)C(C)(C)C(=O)NC)CCC1(C)C c1(OCC(C)C)cccc(C(=O)NC(C)(C)CCNC(C2(C)CC=CCC2)=O)c1 C1(C(N(CCOC)CCNC(c2cc(CO)n(C)n2)=O)=O)CC2OC(=O)OC2C1 Cc1cc(C(=O)NCC2(C)CCCN(C(=O)CC(C)c3ccco3)C2)cc(C)n1 CC(CC(F)(F)F)N=c1[nH]c(N(C)CC2CCCN(C)C2)nc2c1SCC2 C1(C(N2CC3CN(C(=O)C=CBr)CC3C2)=O)CC12CCCc1ccccc12 C12(NC(c3c(C)c(Cl)cnc3)=O)CC3CCC(C1C2)N3C(C1(C)CC=CCC1)=O CC1(C(=O)NCc2ncccc2O)CCCN(C(c2ccc(F)cc2F)=O)C1 CCC(CC(C)C)C(=O)N1CCN(C(=O)CSC(C)C)CC1CS(C)(=O)=O C1(C(=O)NCc2n(C(C)C)cnn2)CCCC(NC(C2(F)CC=CCC2)=O)C1 N1(C(c2[nH]c(=NC)sc2)=O)CCC(C2CCCN(C(=O)C(O)CCC(C)C)C2)C1 O=[N+]([O-])C1CCOCC1OC(c1c(I)ccc(C(F)F)c1Cl)=O N1(C(=O)Cc2ncccn2)CCC(O)(C(N2CC3CC(C2)O3)=O)C1 c1(C(=O)NC)cnn2ccc(C(=O)OC)nc12.c12cccnc1CNS(=O)(=O)C2 Cc1cc2[nH]c(C(=O)NCC3CN(C(c4cn5ncccc5n4)=O)C3)cc2o1 N1(C(C2C(OCC)CC2)=O)CC(C(N2CCN(C(C)(C)C)CC2)=O)C(C)C1 C=C1C(NC(=O)Cc2cc(Br)cc(I)c2)CC2CC1C2(C)C CC#CCCC(=O)NC1CCC(N(C)C(c2nc(OC)c(C)s2)=O)C1 C(=O)(CC(CC)CC)N1CC(C#C)(C(N2CCC2C2CCCCC2)=O)C1 C1(CN(C(C(C)OCCCC)=O)C)CCCN1C(=O)CC1CC1C(F)(F)F N1(C(c2c(C)ccs2)C(=O)NC(C)(C)C)CCC2C(C1)C2(F)F N(C)(S(=O)(=O)N1CC2CC2(C(C)=O)C1)CC#C C1(N(C(=O)C(C)NC(=O)COC)CC)CC(F)(F)C1 C1(C(N2CC(C)C(n3cc(C4CCN(C)C4)nn3)C2)=O)Cc2nccn2C1 CC1=NOC2(C1)CC(C(N1CCCC(CNC(C3CCCCC3(F)F)=O)C1)=O)C2 CCCS(=O)(=O)C(C)C(=O)N(C1CCN(C(=O)COCCF)CC1)CC C(=O)(CC(C(C)(C)C)NC(c1ccccc1)=O)N(CC(O)C1CC1)C C(C(=O)NN=c1cc[nH]cc1Cl)(C1CCOCC1)N(C)C(=O)OC(C)(C)C C1(C(NOCCCC#C)=O)C=CC(NC(c2sncc2C)=O)C1 CN1CC(O)CCC1C(=O)NC(CC(=O)NCCCCc1ncc[nH]1)C1CC1 c1(C(N2C(C)(C)C(NC(=O)CC3CCCOC3)CC2)=O)ccn2nccc2n1 c1(C(N2CCC(C)C(CNC(=O)Cc3cccn3C)C2)=O)ccn2ncccc12 N1(C(c2c(CC)n(C)nc2)=O)CCC(CNC(=O)C(C)=C2CC2)C(F)(F)CC1 C1(C(=O)NC2(CCNC(C(c3scc(C)n3)C)=O)CC2)CN2CCN1C(C)C2 N1(C(c2c(CC)nns2)=O)CCOCC1CC(=O)NCC(C)CC1CCCC1 C1(O)(CNC(c2n(CC=C)ccc2)=O)CCCN(C(=O)C(O)C(F)F)CC1 Cc1cc(C(=O)NCCCC2CCN(C(=O)CC3CC=CC3)CC2)nn1C(F)F c1(C(=O)NC2C(CNC(C(CC)F)=O)COC2)cnc2ccccc2c1 CC(C)(C)C(C(F)F)NC(=O)CC(O)CNC(C1CC2(CCO1)CC2)=O O=C1CC2CC(C(=O)NCC3CC(C(N4CCC(C(F)F)C4)=O)C3)C1O2 c1(C(N2CCCC(N(C(C(C=C)O)=O)CCF)C2)=O)cnc(C)c(C#N)c1 N1(C(C)=O)CCN(C(=O)C(=O)Nc2c3c(cc4c2CCC4)C3)CC(C)(C)C1.C(C)C C(=O)(CCCC(=O)N(C)C)N(CC(CC)NC(=O)Cn1nccn1)CC N1(C(C2C(C)(C)CC2)=O)CCC(N(CCO)C(c2cnc(-c3ccsc3)s2)=O)CC1 Cn1ccc2c(C(N3CCCC(C)(NC(C4CC5CCC5C4)=O)C3)=O)ncnc12 c1(C(=O)NC(C2CCN(C(C3(C(C)C)CC3)=O)C2)C)cc(F)c(N)c(F)c1 C(=O)(CC(C)(C)N(C)C(c1cc(OC)nn1C)=O)N(CC(C)O)CC N1(C(CC=C)=O)CC(CCNC(c2cc(Cl)cn2C)=O)C(C)C1 CC(C)CCC(F)C(=O)N1CCCCC(C(=O)NCC2CC3CCC2O3)C1 c1(NC(C)=O)ccc(C(=O)NC2(CN(C(=O)CN(C)C(C)=O)C)CC2)cc1F N1(C(C(C=C)O)=O)CCC(NC(c2c(C)cc(C)cc2N)=O)C(CO)CC1 c1(C(C)OC)nc(C)c(C(=O)NC2C=CC(CNC(=O)CCn3cnnn3)C2)s1 N1(C(CNS(NC)(=O)=O)=O)CCC(CNC(c2ccc(Cl)o2)=O)C2CC12 C12(C(=O)Nc3cc(C)sc3)CC(CCO1)N(C(C1CC13CCCC3)=O)C2 c1(C(=O)OC)cc(S(=O)(=O)N2CCN(c3[nH]c(=N)ccc3Br)CC2)ccc1I C(=O)(C1=CCOCC1)NCCC(=O)NC1CC1.CC1CCCC12C(=O)N2 c1(C(=O)NCC2(CC(=O)OC)CCCC2)cnccc1Cl CC(C)C(C)CCNC(c1cn(C2CCC2)nn1)c1nnnn1CCCSCCO N1(C(C2C(C)OC(=O)N2)=O)CCCC(NC(c2ncccc2F)=O)CC1 c1(C(=O)NCCN(C)C(C2CC3(C2)CC2(CC2)C3)=O)sccc1S(N)(=O)=O c1(C(N2CC3C(NC(c4c(C)coc4)=O)CC(C3)C2)=O)cc2cc(F)ccc2s1 C(=O)(CC(O)CC(C)(C)C)N(CCC)CCNC(c1c[nH]c(C)c1)=O c1(CSC)ccn2ccnc2c1.N12CC(C1)C(=O)N1CCC1CNC2=O C=Cc1cncc(C(=O)NC2(CO)CN(C(c3ccnc(OC)c3)=O)C2)c1 C1(CNC(C(C)n2ccnn2)=O)CC2(CCN(C(=O)C3=COCCO3)CC2)CO1 C#CC1(O)CCCN(C(C2(C)CN(C(=O)C(CO)NC(N)=O)C2)=O)C1 C(C(C)(C(=O)NC1CCC1C(=O)NCC1CC(C#N)C1)OC)OC c1(C(N2CCC(CC(C)C(=O)OCc3ccccc3)CC2)=O)c(Br)cncc1Br C(C)(CNC(=O)C(c1cnn(C)c1)OC)(CC(C)C)NC(C(CC=CCC)C)=O C1(c2n(CC)nc(Cc3nc(-c4ccc(Cl)c(Cl)c4)cs3)n2)CC12CCOCC2 C#CCCC(O)CCNC(C1CC(O)CN1C(=O)COCCCN(C)C)=O N1(C(C2C(=C)CC2)=O)CCC2CN(C(=O)CC3CCC4CC4C3)CC2CC1 CC1OCCC1C(=O)NCC1CC(C(=O)N(C)CCC2CCCCC2)C1 CCCCS(=O)(=O)N1CCCC1C(=O)NCCNC(=O)CCOC1CCCCC1 c1(C(=O)NCCC2(OC)CN(C(C3CCC(C)C3)=O)C2)cnc(C(C)C)nc1 Cc1c(C(N2CCC(O)(CNC(C3(n4cccn4)CC3)=O)C2)=O)c[nH]c1C#N N1(C(C(CC(C)C)(C)C)=O)CC2CCC1C1CN(C(=O)CCc3cncs3)CC21 C1(C(N2CC(CCC)C(CO)C2)=O)CN(C(c2cscc2Cl)=O)CCN1C C(CCN(C(=O)CSS(C)(=O)=O)C)(C(C)C)NC(C(C)NC(CC)(C)C)=O c1(CNC2C(n3cc(CC(C)C)nn3)CC2)ccc(S(=O)(=O)NS(C)(=O)=O)cc1 n1(CC)c(CCCNC(=O)NCc2sccc2C)nc2ccccc12 Cc1cc(C(=O)NCC2CCC2NC(=O)CC(c2c(C)n[nH]c2C)C)sc1C CC1CCn2ncc(C(=O)NC(C)CNC(c3nc4cccnc4s3)=O)c2C1 n1(CC)cc(Cl)cc1C(=O)N(CC(CO)(CO)NC(=O)Cc1cnc[nH]1)C CC1(C)C(NC(=O)CCCN2CCCC2)CCN1c1nccnc1F N1(C(CCC=C)=O)CCCCCC1C(=O)NCCC1CC1C c1(C(N(C)CCN2CCN(C(=O)CCOC3CC3)CC2)=O)ccn2nccc2n1 CC1(C)Cc2cc(C(=O)NCC3C4CN(C(=O)CC5CCOC5)CC34)ccc2O1 c1(C(C(=O)N(CC(=C)C)C2CC2)N2CCC2C2CCC2)n[nH]cc1Br c1(CN2CCN(C(c3cc(Cl)ncn3)=O)C3C2C3)n[nH]c2c1CCCCC2 CCCCC(CNC(=O)C(C(C)C)NC(=O)OC)NC(=O)CN1CC(C)(OC)C1 CC(C)CC(C)(O)C(=O)N1CC(NC(=O)C=Cc2cncnc2O)CC(F)C1 C(=O)(C1CCCc2c[nH]nc21)N1CC(CNC(c2c(CC)cncc2)=O)C1 C(N(C)N1CCC2CC(C1)CC(C(=O)OC)(OC)C2)c1cccc(Cl)c1 N1(CC(=O)NC(c2n(CC)ccn2)C)C(=O)NC2(CCC(C)CC2)C1=O S(=O)(=O)(c1cnc(Cl)nc1)NC1CN(C(c2c(Cl)ccc(F)c2F)=O)CC1F N1(C(C2(CC)CC2(F)F)=O)CC=C(CCNC(c2ccc(OC)c(C)c2)=O)CC1 CC1CCN(C(=O)C2=NNC(=O)C2)C(CNC(C2COC(=O)O2)=O)C1 c1(C(=O)NCCC(CNC(c2ccc(OC)c(F)c2)=O)O)c(C)cc(=O)oc1C S(=O)(=O)(CCC(=O)N1CCC(CO)(NC(=O)CN2CC3CCC2C3)C1)N(C)C N1(C(c2cccn3c(Br)cnc23)=O)CCCC2C1CCN2C(=O)C(F)F C1(C(=O)NCC2(NC(c3[nH]c(=NC)sc3)=O)CCC2)CC(C)(C)SC(C)(C)C1 N1(C(c2cn(CC(C)N)nc2)=O)CC2COCC2(C(=O)N(C)C)C1 C1(CN(C(=O)Cc2ccc(F)cn2)C)CN(C(C2CC(N3CC(O)C3)C2)=O)CC1O N1(Cc2cn(C)nn2)CC2(CCN2C(=O)Cc2cc(Br)cs2)C1 C(C(C(F)(F)F)C(F)(F)F)c1nn(C2CCCN(C)C2)c(-c2cccc(Cl)c2)n1 C1(NC(CCCOCCOC)=O)C2CCC(C2)C1C(=O)NC1CCCC(O)C1 C1(C(N(CCOC)CCNC(c2nn[nH]c2Cl)=O)=O)C2CCC1CC2 N1(C(C(CCC)F)=O)CCCCCCC1C(=O)NC1CCCCC1(C)C Cc1ncnc2c1CC(C(=O)NCCC1(NC(=O)CC(F)F)CCCC1)CC2 N1(C(C2C(CN(C)C)CCC2)=O)CCN(C)CC1CNC(c1cnncc1O)=O C1(CNC(C=CC=CC)=O)CCCCN1C(=O)C=CC1CCCC1 c1(C(N(C(c2sccc2C)C(=O)NCCCSC)C)C)cccc(O)c1 N1(C(=O)CCc2cccnc2Cl)CCN(C(c2cc(CO)on2)=O)C2(CCC2)C1 Cc1c(C(=O)NC2(CNC(c3cnn[nH]3)=O)CC2)ccc2c1CCC2 N1(C(c2cnc(OCC)s2)=O)CCCCCC(NC(=O)CC2CCOC2(C)C)C1 c1(OC)ccc(C(=O)NC(C2CCN(Cc3cccs3)CC2)C)nn1 CCCCCC(CC)C(=O)N1CCC(CCC(N2CCc3nocc3C2)=O)CC1 C1(C(=O)NC2CC(C(=O)OCCNC(C3C(C)CN(C)C3)=O)C2)CC(C)(C)CN1C O=C1NCc2c(C(=O)NCC3CC(F)CN3C(c3cnn(CF)c3)=O)cccc21 C(CC(C(=O)N1CC(CCNC(=O)C=C2CCC(C)C2)C1)OC)NC(=O)OC CCCCC(CC)NC(=O)CNC(=O)C(CC)OC c1(C(N(CC(CC)NC(=O)COc2ccccc2)CC)=O)nnn(C)c1N C1(C(=O)NCC(CCC)OC)CC(O)CN1C(=O)CCc1nncs1 c1(OC)cnc(C(=O)NC(Cn2cncn2)C(=O)NC2(C3CC3)CC2)cn1 N1(CC(C)C)CC(C)N(c2nnc(C(=O)N(C)C)n2CC2(C)CCCO2)CC1C N1(C(C(C(C)C)NC(C)=O)=O)CCC2(CC1)CN(C(C1COC(=O)O1)=O)CCO2 C1(N(C(c2n(C(C)C)nnc2)=O)C)CCCN(C(C2C(C#N)C2(C)C)=O)C1 c1(OC(c2cc(C)on2)C)nc2ccccc2[nH]1 c1(C(N2C(C3N(CCCCCOC)CCC3)CCCC2)=O)cc(C2CC2)nc(O)c1 Cc1c(I)c[nH]c1C(=O)NCCNCCCOCc1ccccc1 Cc1nc2c(C)cc(C(N3CCC(NC(=O)C(O)CN(C)C)C3)=O)cn2n1 CCC(CC)CCC(=O)N1CC(NC(=O)CCC2(C)CC2)CC1(C)C C1(CC(=O)NCCCN(C(C)C)C)CN(C(C2CCC3(CC3)C2)=O)C(C)(C)C1 CCC(C)C(C(=O)NC1CCCCCC1)N(CC)Cc1ncnn1C(C)(C)C Cc1cccc(C)c1C(O)C(=O)NC1CCC(NC(C2CC(N(C)C)C2)=O)C1 N1(c2nnc(N3CCC(COCC)C3)s2)CCC(C(C)(C)C)CC1 N1(C(c2c(CCC)n(C)nn2)=O)CCCN(C(=O)CCC=C(C)C)CC1 C#CC1(C(=O)NC(C)C(C)(C)CC)CCN(C(=O)COCC(F)F)C1 c1(C(=O)NC2CC(C)(NC(Cc3c(C)occ3)=O)C2)ccccc1S(C)(=O)=O c1(C(N(C)CC2(O)CCN(C(CCSCC)=O)C2)=O)cc2c(cnn2C)nc1C c1(C(=O)NCCC(C)NC(C=CSC)=O)cccc(Cl)n1 N1(C(C(n2cc(Br)cn2)C)=O)CCCC(n2cc(-c3cnc(Cl)s3)nn2)C1 N1(C(CSCC(C)C)=O)C2CCCC1CC(CNC(c1ccc(N)c(F)n1)=O)C2 Cc1n[nH]c(C)c1C(=O)NCCn1cc(C(N2CCCC3CC23)=O)cn1 N1(C(CCc2c(C)cccc2)=O)CC(CNC(=O)Cc2ccon2)N2CCC1C2 c1(C(n2cc(CNC(c3nccc(NC)c3)=O)nn2)C)ccc(Br)cc1C C1(CC(=O)NCC2CCN2C(c2nocc2Cl)=O)NC(=O)NC1=O c1(C(N2CC(NC(c3ccn(C)c3)=O)C2)=O)cccc(C2=CCOCC2)c1 CS(=O)(=O)c1cc(S(=O)(=O)NNC(=O)C2OCCC2c2ccccc2)cs1 N1(C(C(C)=C2CCC2)=O)CCCC(C2CCN(C(c3cc(C)cc(N)c3)=O)C2)C1 c1(C(C)O)ccc(NC(=O)C=C2CCN(C(c3ccc(OCF)cn3)=O)CC2)cc1 C12(CNC(CN(C(C(C)C)=O)C)=O)CC1CN(C(c1ccn(C)n1)=O)C2 C1(NC(CCCCN(C(CC2ON=C(C)C2)=O)C)=O)CC2C(C1)C2(F)F C(=O)(C(CC(C)C)SC)NCC(Sc1ncccc1SC)NC(C(OC)SC)=O C(=O)(C(O)CC(N)=O)N(CCCNC(=O)C(=O)NCc1ccc(F)cc1)C(C)C C(=O)(C(C)(C)C(N)=O)NCCC1(O)CCN(C(c2noc(C)c2Br)=O)C1 C(CNC(=O)C(c1ccccc1Cl)(F)F)(C(C)C(C)C)NC(C1(CC)CCC1)=O C1(NC(C2CC=CC2)=O)CCN(Cc2ocnc2Cn2cc(COC)nn2)C1 CC1CN(C(C2CC2(Cl)Cl)=O)CC1n1cc(-c2cncc(C(=O)O)c2)nn1 Cc1cc(C(=O)CN2CCC(C(=O)N=c3cc[nH][nH]3)C(c3cccs3)C2)c(C)n1CC(C)C N1(Cc2c(OC)ccs2)CCC(O)(C(=O)NCC(N2CCOCC2)=O)C1 C1(NC(c2c(C)ncs2)=O)CCCC(NC(=O)C=CC2CCCCCC2)CC1 C1(C(CNC(=O)CCc2cccs2)NC(C(C)O)=O)CCCCC1 N1(C(CC=C(C)C)=O)CCCC(N(C(=O)CSCC(F)(F)F)C)C1 Cc1c2cc(C(=O)NCC(C(N)=O)N(c3ccccc3)C)ccc2nn1C c1(C(N2CC(N(C(c3cc(OCC)no3)=O)C)C(F)C2)=O)nn(C)c2c1CCC2 C1(C(=O)OCC2CCC(C(=O)OC)O2)CN(C)CC(C)O1 C#CC1(C(=O)NCC(C)(O)C(C)(C)C)CCN(C(=O)CC(C)(C)CN(C)C)C1 N1(C(c2nc(C(C)OCC)sc2)=O)CC(OC)CC(C)C1.C12(CCC1)C(=O)NC2 C12(C(=O)OCC)CCC(CN(C(=O)CC3(C(=O)O)CC3)C1)C2 N1(C(C(CCC)N(C)C)=O)CCN(C)CC1COC1(C(=O)NC)CC1.C(C)(=O)O S(=O)(=O)(CC(=O)NCC(O)CNC(C1(CC2CCCC2)CCCC1)=O)N(C)C N1(C(c2ccccc2)C(=O)NCC#C)CCCC(C)C1CCO C1(CNC(=O)C(F)C2CCOC2)COCCN(C(c2cn(CCO)nn2)=O)C1 C(CO)(CCCNC(c1csc(C)c1C)=O)NC(CCN(C(CCC)C)C)=O C(=O)(C(F)(F)C(F)F)NC1C(NC(=O)Cn2nnc(-c3ccco3)n2)CCCC1 c1(N2CC(C(=C)C)C2)nc(N2CCCN(C(C)CO)CC2)nc2c1CCCCC2 C(=O)(C1CCCc2ncccc21)N1CCN(C(C=CCC)=O)C(C)C1 N1(C(CCNC(COC)=O)=O)CC(CNC(=O)CC2CC3CC3C2)C(F)(F)C1 CCCC(C(=O)N1CCN(C(=O)C(C)CC(F)(F)F)C(CCOC)C1)S(N)(=O)=O C12(C(=O)OC)CC1CN(C(=O)C(C1CN(C(=O)COc3ccc(C)o3)C1)OC)C2 C(=O)(CC(O)C(C)C)N(CCNC(CC(c1c(C)cccc1)C)=O)C1CC1 c1(NCc2nccc(C)n2)ccc(S(=O)(=O)NCCC2CCC(C)C2)cc1Br C(=O)(C(CNC(c1cnc(OC)nc1)=O)C(C)(C)C)NC(CC=C)CC c1(C(=O)NCC2(F)CCC(NC(C(COCC)C)=O)C2)c[nH]c2nccc-2c1 C1(C)(C(=O)NC(CSC)C)CN(C(c2csc(C)n2)=O)CC1C c1(C(=O)NC(CC=C)CNC(c2ccc(C(N)=O)cn2)=O)cc2cc(Cl)sc2[nH]1 C1(C(=O)OC)CC2(CC(NC(=O)CC3(C)CCNC3)CCO2)C1 N1(C(C(C)OCC=C)=O)CCN(C)CC1CNC(=O)CCc1ncc(C)[nH]1 C1(NC(CNC(=O)CNC(C2CC=CCC2)=O)=O)CCOC2(CCC2)C1 CCC(CC)C(C(=O)NCC1(C(N2CCC(C)(NC(C)=O)C2)=O)CC=CC1)OC c1(-c2c(OCCC)cccc2F)cc(S(=O)(=O)NC(C)CO)c(C)cc1C c1(N2C(C3CCN(C(C(COC)O)=O)C3)CCC2)ncnc2cccnc12 N1(CCC#C)CCCC(CNC(=O)C(=O)NCC(c2ccccn2)(F)F)C1 N1(C(C(C(C)C)C)=O)CCC(C2(NC(C3CCC(F)CC3)=O)CC2)CC1 c1(C(C(=O)NC2CCOCC2)N(C2CCCC2)CCC)ccc(F)cc1C N1(C(C(C)(C)C)=O)CCCOC(CNC(C2(c3ccccc3Cl)CC2)=O)C1 c1(C(=O)NCC2N(C(c3cc(OC)n[nH]3)=O)CCOC2)cncc2c1CCC2 Cc1cccc(CCC(N2CCN(CC(N3CCC(C(C)(C)O)C3)=O)CC2)=O)c1 CC1CCN(C(c2cccn2C2CC2)=O)CC1NC(=O)Cc1cc(Cl)n(C)n1 C(CNC(=O)OCC(C)C)(CC(=O)N1CCC(OC(=O)N(C)C)C1)OC C(=O)(C(CCF)NC(c1cc(C)c[nH]1)=O)N1C(COC)CCC1 C(C(CNC(=O)C(C)(F)CC)C(F)(F)F)NC(c1n(CC)ccn1)=O C1(CC(=O)NCCN(C(=O)COCc2cnn(C)c2)CC)CCCCC12CC2 N1(C(CNC(C2C(COC)CC2)=O)=O)CCC(N(C)C)C(C)C1 CCC(C)(C)CC(=O)N(C1CCCCCC1)CCNC(c1cn(C)nc1SC)=O c1(C(N2CCC(C(C)Nc3nccc(C(F)(F)F)n3)C2)=O)ncc2c(n1)COC2 c1(C(=O)NCC(CNC(c2nn(CC)c(C)c2)=O)CO)ccc(F)c(C)c1 C1(OC)C=CCN(C(=O)C=CC(C)NC(C2(C)CCCC2O)=O)C1 c1(C(N2C(C)CC(CNC(c3ccsc3)=O)C2)=O)cc(Cl)c(F)c([N+](=O)[O-])c1N c1(C(N2CC(c3cn(CCC)nn3)(C(=O)OC)C2)=O)c[nH]c2cc(F)c(F)cc12 C(=O)(C(=O)CC(C)C)NCC1C(C(N(CCO)Cc2ccc(C)cc2)=O)C1(C)C Cn1cc(Br)c(C(N2CCCC(OCc3cn(CC4CCC4)nn3)C2)=O)n1 CC1CCN(C(=O)CC2CCC3CC23)CCN1C(c1ccc(N2CCC2)nc1)=O C12(C(=O)OC)CC(CNC(=O)CN(C)C(=O)OC(C)(C)C)(C1)OC2(C)C c1(C(N2CC(C#N)C(NC(C3CCCCC3)=O)C2)=O)c(Cl)ccc2c1OCO2 c1(C(N2CCCCC2CNCc2ccc(Cl)s2)=O)cc(Cl)cc(Cl)c1 c1(CC)ccc(CC(=O)NC23CC2CN(C(=O)CC2COC(=O)C2)C3)cc1 C1(NC(c2ccc(OCC)nn2)=O)CCC12CCN(C(=O)C(N)=O)CC2 CCC(C)CCCC(=O)N1CC(C)(C)CC1CC(=O)Nc1ccc2c(c1)OCO2 CC(C)C(C(=O)NCCCc1nccs1)N1CCCCCC1 c1(CCCC(=O)NCC2(O)CN(C(C(C=C)(C)O)=O)C2)ccc(C)c(C)c1 C1(NC(c2ccoc2Br)=O)CN(C(=O)CC2CCCCC2O)CCC1C(F)(F)F C1(NC(C=NOC)=O)CCC2(CC1)CC(NC(=O)C=CC(N1CCCCC1)=O)C2 CCCC(C)(CCC)C(=O)N1CCOC(C(N2CCC(CC(C)O)CC2)=O)C1 C1(CC(=O)N(C2CCCC2)CCNC(C2CC2CF)=O)(OC)CCOCC1 C1(CNC(=O)C=Cc2cc[nH]n2)CC2(CCC2)CN1C(c1ccccc1Cl)=O c1(CNC(CC)=O)cc(C)c(C(=O)NC(C)(C)CC2CCCC2)o1 Cc1ncc(C=CC(N2CC3CC2C3CNC(=O)CSCc2ccncc2)=O)s1 C1(C(N(C2CN(C(CCC(C)C)=O)CC2O)C)=O)CCCC1C1CC1 N1(C(c2cc(Cl)c(Br)[nH]2)=O)CCN(C(=O)C(F)CC2CCC2)C(CO)C1 C1(C2CCCC2)(C(N2CC(C(C)NC(c3cc(Br)c[nH]3)=O)C2)=O)CCNC1=O C1(CNC(CCNC(COC)=O)=O)CCC2CN(C(=O)C(F)(F)C(F)F)CC12 Oc1nc2nc(-c3nc(CSC4CCC4)nn3CCc3ccccc3)ccc2[nH]1 N#Cc1c(NCCNC(=O)Cc2ccc3c[nH]nc3c2)ncc2c1COCC2 CCC(C(=O)N(CC(C)N(C(=O)CC1(COCC)CCC1)C)C)N(C)C n1(C(C)C)cc(C(=O)NCC(c2ccccc2)NC(c2cnco2)=O)ccc1=O C1(CC)C(NC(C2CCCC2(C)C)=O)CCCN1C(=O)COCCN(C)C C1(NC(C2(CCOCC)CCC2)=O)CCN(C(=O)Cc2csc(S)n2)C1 c1(C(N2C(C)(CNC(C3CC(CCO)C3)=O)CCC2)=O)cc(F)cc(F)c1 c1(C(N(C)CCOCCN(C)C(C2CC2CF)=O)=O)ccc(S(N)(=O)=O)cc1N N1(C(C2(CNC(=O)CCn3cccc3)CC2)=O)CC2C(C1)C2(F)F C1(C(F)(F)F)(Oc2ccccc2)CC2CCC1CC2.C1(=O)C#CC2CN(C2)C(=O)N1 c1(C(N2C(CNC(C(C)N(C)C)=O)CC2)=O)c[nH]nc1-c1ccccc1 c1(C(=O)NCC(O)CNC(C23CCCCC2C3)=O)ccc2nccnc2n1 c1(-n2cc(CN(C)C(C3CCCOC3)=O)nn2)ccc(-c2ccc(F)cc2)cc1 C1(NC(C(N2CC(C)C2)C)=O)C(C(=O)NC2CN(C(N)=O)C2)C1(C)C CC1C(C(=O)OCC2(c3cccs3)CC2)N1CC(=O)N(C)C N1(C(C(C(CC)C)O)=O)CC2CCC(NC(=O)C(C(C)C)OC)CC2C1 NC1CCC(N2CCN(C(=O)C(N3CCC(c4ccncc4)C3)=O)CC2)CC1 CC1CCN(C(C2(C)CCNC(=O)C2)=O)CC1CNC(=O)Cn1nccn1 c1(OC(C(=O)NC2CCN(C(c3c(C(C)=O)ccs3)=O)C2)C)ccc(C)cc1C C1(NC(c2cc(C)nnc2)=O)CN(C(=O)CN2CC(C)C2)CC1C1CC1 c1(OC)ccc(C(=O)N(CCC(C)NC(c2coc(C)c2)=O)C)c(OC(C)C)c1 C1(COC)CCCCN(C(c2cc(C3CC3)nn2-c2ccccc2)=O)C1 c1(CN2CCCC(C=C)C2)cc(=NCC2CCCC(C)CC2)[nH]c(C)n1 c1(C(=O)NCC2(NC(=O)CC3(O)CC3)CC2)ccc(CN2CCSCC2)cc1 C1(NC(C#CC(=O)O)=O)CC2CCCC(C1)N2Cc1cc(F)c(F)c(Cl)c1F c1(CNc2ccc(C=CC(=O)Nc3c(C)cnc(O)c3)cc2)cc(Cl)c(O)cc1O Cc1cc(C(=O)N(C)CC2(O)CN(C(C3(C)C=CCC3)=O)C2)cc(N)c1 c1(CNC(CSC)=O)ccc(C(=O)NCC2(Cl)CCC2)cn1 c1(C(N(CCNC(c2c(C#C)cn(C)n2)=O)C)=O)c(F)cccc1[N+](=O)[O-] c1(C(C(=O)NC2C(NC(c3cc(F)ccc3Cl)=O)C2)O)ccc(F)cc1F c1(CN(C)C(=O)NC2CC(C(=O)O)C3CC23)nn(C)c2ccccc12 C1(NC(C(=O)NCCOc2cccc(C#C)c2)=O)CCc2cc(OC)ccc2C1 N1(C(C(CC)(C)C)=O)CCCC2(CCN(C(C3(F)CCCC=C3F)=O)C2)C1 O(CP(C)(C)=O)NCCC(=O)NC(C)CNC(=O)CCSc1nnnn1C N1(C2C(NC(C)=O)COC2)CCN(C(=O)C(=Cc2cccnc2)F)CC1 CC(CC(=O)NC1CCC2CC1CN2C(C1CCN(C)CC1)=O)CC(C)(C)C N1(C(c2c(C)n(C)cc2)=O)CC2CCC(CNC(C3CCOC3C3CC3)=O)(C2)C1 C1(NC(C(CCC)NC(C)=O)=O)(CO)CCCN(C(=O)CSc2cccs2)C1 C(=O)(C(F)(F)COCC(=O)NC(C)C)Nc1c(OC)c(C(N)=O)ccc1 C1(O)(CNC(C(C)=CC=CC)=O)CC2CCC(C1)N2C(=O)C(C)Cn1ccc(C)n1 N1(C(C(F)=CCC)=O)CCc2ccccc2C(NC(=O)Cn2ncnn2)C1 CC1CC(C(=O)N(CCCn2ccnc2)C)CCN1C(C1CC(O)CN1C)=O N1(C(c2ccn(CCF)n2)=O)CCN(C(c2cccc(Cl)c2F)=O)C2CC12 N1(C(=O)CC2CC(C3CC3)C2)CC2CN(CCO)CC2C1 C1(O)(CNC(C(COC)C)=O)CCN(C(c2ccc(=O)n(O)c2)=O)CC1 C(=O)(C1=NOC2(CCC2)C1)N(C(C)(C(N1CCCC(O)C1)=O)C1CC1)C c1(C(=O)NCC2CC(N(C)CC)C2)ccccc1SCCO CC1(CNC(c2csc(Cl)n2)=O)CN(C(=O)Cc2cccs2)CCO1 C(CN=c1nc(C2CC2)[nH]c2c1CCC2)NC(C1CC12CC2)=O c1(C(C)=O)ccc(C(=O)NCC2(CN(C(=O)Cc3csc(NC=O)n3)C)CC2)[nH]1 c1(C(=O)OC)c(NC(=O)Cc2ncn3c2CCC3)ccc2c1CCCC2 C1(CNC(c2c(SC)cccc2F)=O)CC2(CCC2)CN1C(=O)Cn1cccn1 C12(C(=O)NC(C=C)(C)C)CCCC1CCN2C(=O)CCCOC C1(C(C)(C)C)(CNC(C2(C)C=CCC2)=O)CCN(C(c2ccc(C(N)=O)o2)=O)C1 CCCCC(F)C(=O)NCC(CC(=O)N(C)Cc1nccn1CC)OC C(=O)(C(F)(F)C(C)(C)O)N1CCC(C(C)NC(C2CCC3(CCC3)CC2)=O)C1 Cn1cc(C(=O)NCCNC(C2CCCC(CF)C2)=O)c(Cc2ccccc2)n1 N1(C(C(C)NS(C)(=O)=O)=O)C2CCC(C2)C1CNC(=O)CSc1ccccn1 C1(C)(C(N(C(C)C(=O)NC2CC(CCSC)C2)CCC)=O)CCCC1 C1(C(N2CCC(CN(C(=O)CNC=O)C)C2)=O)CC12CCC1(CC1)CC2 N1(C(c2cn(CCNC(CC(C=C)(C)C)=O)nn2)=O)CCC(CO)=C(F)C1 C1(CC(=O)OCC)CCC(C(=O)NC2CCCN(Cc3cc(C)[nH]n3)C2)CC1 Cc1nc(-c2ccc(Cl)cc2)cc(=NCCOc2cnc(Cl)c(Cl)c2)[nH]1 N1(C(C2(C(N)=O)CC2)=O)CCN(C(c2coc(O)n2)=O)C(CN2CCCC2)C1 Cc1sc2cc(F)ccc2c1CCNC(C1CCCC(P(C)(C)=O)C1)=O S(=O)(=O)(c1cccc(C(N2CC(c3c(F)cccc3F)(O)C2)=O)c1)N(C)C CN1CC(O)CC1(C)C(N1CC2(C1)CN(C(C1CC1(C)Br)=O)C2)=O c1(CC(=O)NC2C(NC(C=CCC)=O)CCCC2)nnc(O)nc1O c1(NC)ccc(C(N2CCCCC2C(=O)NC(c2cnc[nH]2)C)=O)cc1 C1(C)(CC(=O)N(C(=O)CCNCC)CCC)CC(F)(F)C1.S(=O)(=O)(CC)N CCC(C)C(O)C(=O)NCC(CCOC)NC(=O)Cc1ccc(C)c(OC)c1 Cc1c(Br)c(C(=O)NCCCN(C(=O)C(c2cnccn2)C)C2CC2)nn1C c1(-c2scc(CN(C(=O)CC3CCCSC3)C)n2)ccc(F)cc1 N1(C(C2C(C)C2C)=O)CCc2c(CNC(C3(F)CCCCC3)=O)cccc2C1 C(c1ccc(F)cc1[N+](=O)[O-])=CC(=O)NC1CC(CNC(C(C#N)C2CC2)=O)C1 c1(C(=O)NCCC(C(=O)N2CCC(C(=O)NCC)C2)OC)c[nH]c2ccccc12 c1(NC(C2(C)CCN2C(c2cc(O)nc(O)n2)=O)=O)c(Br)cc(F)cc1[N+](=O)[O-] C12(C(N3CCCCC3c3cn[nH]c3)=O)COC(C1)C(NC(=O)C(F)(F)CO)C2 CC(C)(C#N)CCC(=O)NC1CCCC1NC(c1scnc1C1CC1)=O N1(C(Cc2cccc(OC)n2)=O)CCC2(NC(c3ccc(C4CC4)o3)=O)CC2C1 C1(=O)CCOCCCN1.C1(C(C)C)CC1C(=O)N(C)CCC1CC1 Cc1cc(C(N2CC(c3ccccc3)CC2C(=O)NC2CS(=O)(=O)C2)=O)n(C)n1 c1(CC(=O)NCC(CC=C)NC(C2(C)CCCCC2)=O)ccc2ccoc2c1 c1(C(=O)NCCN(C(C(C)SC)=O)CC(C)O)cccc2ccncc12 Cc1cn2c(CC(N3CC4(CCC4NC(C4CC45CCCC5)=O)C3)=O)csc2n1 C1(C(=O)NCCC2(CNC(c3c[nH]c(=N)s3)=O)CC2)CSc2ccccc2O1 Cc1cccc2cc(C(=O)NC3CC3CNC(=O)C(C(C)(C)C)C3CCC3)oc12 N1(C(c2scc(OC)c2)=O)CC2CC2(NC(=O)CC2CCCN(N(C)C)C2)C1 N1(C(C(CCC)N(C)C)=O)CC2CS(=O)(=O)CC2(NC(c2cn(C)[nH]c2=N)=O)C1 C(CC(=O)NC1CCCC(O)C1)(C(F)(F)F)NC(c1cc(C)cc(C)n1)=O c1(C(=O)NCC(C)(C)NC(C(C)NC(CC)=O)=O)ccc(-c2cccs2)[nH]1 c1(N2CCN(C)C(=O)CC2)ccc(S(=O)(=O)NCC2(F)CCOCC2)c(Cl)c1 CC1(CNC(c2cc(Cl)cs2)=O)CCCN(C(=O)C=CC2COC(C)(C)O2)C1 c1(C(=O)NC(C)CN(C(=O)CCNC(N)=O)C)nc[nH]c2nccc1-2 N1(C(c2nnn(C)c2N)=O)CC(C(=O)NC2CN3CCCC2C3)CC1(C)C CCCS(=O)(=O)C(C)C(=O)NC1CCN(C(c2cccc(NC(=O)NC)c2)=O)C1 Cc1cc(C(N2CCC(C(C)(C)NC(C3(C4CCCO4)CCC3)=O)C2)=O)c(C)s1 c1(OC)cnnc(C(N2CC(CC(C)(C)CNC(=O)CSCC(F)(F)F)C2)=O)c1 N1(C(C(CC(C)C)ONC(=O)Cn2cc(Cl)cn2)=O)C2CCC1CC1(C2)N=N1 N1(C(c2c(COC)noc2)=O)CCCC2CN(C(c3nncs3)=O)CCC12 c1(OC)c(C(=O)NC2CCC(CCNC(c3[nH]ncc3C#N)=O)C2)cccc1Cl N1(C(C2CC(=C)C2)=O)CC2C(C1C(=O)Nc1ncccc1C(=O)NC)C2(C)C S(=O)(=O)(c1cnc(N2CCC(C)(CS(C)(=O)=O)C2)c(Cl)c1)NCCCSCC N1(C(c2ccn(C(C)C)n2)=O)CCC(C(=O)NCCc2ccccc2F)(CF)C1 N1(C(C2C(C(=O)NCC3CC3)C2)=O)CC2CNC(=O)C2C1.c12ccc(cc1)[nH]c2=O c1(C(N2CC(C)C(CCNC(C3C=CCC3)=O)C2)=O)nc(Cl)ccc1N C1(NC(c2n(CC)ccn2)=O)C2CN(C(=O)C(C3CC3)OC)CC12 C1(CNC(CN(C(=O)OCC)C)=O)CC(NC(C2CCN(C)CC2)=O)C1(C)C C1(C(N2CC(C)(C(N)=O)C2)=O)CC2(CCC2)C1.Cn1nccc1C1C(=O)N1 N1(C(C2(CCNC(C(CC)(C)OC)=O)CC2)=O)CC(C)C12CCOCC2 N1(C(c2ccc(Br)cc2F)C(=O)NC(C(=O)OC)C)CC2(C)CCC2(C)C1 N1(C(C(=O)NC2CCOC2)CC2CC2(Cl)Cl)CCC2(CC1)CC2(F)F c1(NC(C2C=CC(NC(c3c(C)n[nH]c3)=O)C2)=O)ccccc1NS(C)(=O)=O CC1CCC(C(=O)NC(c2ccccc2)(C)C)CN1CCCc1ccccc1Cl C1(C#N)(NC(c2c(C)nn[nH]2)=O)CCN(C(c2cccc(I)c2O)=O)C1 c1(C(N(CCN(C(=O)CC2(O)CCOC2)CC)CC)=O)cnn(CC)c1C c1(NC(C2N(Cc3c(C)cccc3)CC(F)(F)C2)=O)cccn2ncnc12 c1(C(=O)NCC2(OC)CN(C(C(C3CC3)OCC)=O)C2)ccnc2c1cnn2C N1(C(c2ccc(C(C)=O)o2)=O)CC2(C)CC1(C(=O)N(C1CCC1)CC1CC1)C2 c1(C(N(CCOC)CCNC(C2CCC2F)=O)=O)cccc(N(C)C)c1 N1(C(c2[nH]ccc(=N)n2)=O)CC2CN(C(C3(F)CCOC3)=O)CC2C1 CCC1=NOC(CC(N2CC(O)CC2C(=O)N(C)CC2CC2(C)C)=O)C1 c1(NC2CC(=C)C2)ncc(C)cc1S(=O)(=O)NCc1cc(Br)ccn1 CC(CN(C)C)CCC(=O)N1CCC(NC(C2CN(C3COC3)C2)=O)C12CC2 c1(COC(C(=O)N(CC(CC)NC(C2(C(N)=O)CC2)=O)C)C)ccc(C#N)cc1 c1(NC2C3(CC(OC)C3)C2)nc(NC(C)CC(N)=O)c2cnn(C)c2n1 c1(C(=O)OC)c(C)cc(C)nc1NCC1CCCN(C(c2c[nH]cc2Br)=O)C1 Cc1cc(N)ccc1C(N1CC(C)(C)CC1CNC(=O)CC1CC(=O)NC1=O)=O C1(CNC(c2c(C)scn2)=O)CN(C(C2CC(O)(C(F)F)C2)=O)C2CCN1C2 CCCCCCC(=O)NCC1(NC(=O)CCc2nccn2C)CCCCC1C c1(NC(N(C)Cc2cc(C)no2)=O)ccc(NS(=O)(=O)C(C)C)cc1 c1(N2C(=O)CC(NC(c3c(N)cc(Cl)cc3Cl)=O)C2)ccc2c(c1)OCCCO2 n1(CC(=O)Nc2cc(C)c(F)c(C)c2)ccc(=NCc2cnco2)nc1O N1(C(C2C(C=C)C2)=O)CC2CCN(C(=O)CCOc3ccccc3)CC2C1 N1(C(C2(C)CC(C)C2)=O)CCN(C(=O)C(c2ccn(C)n2)C)C(CO)C1 Cc1cccc2c1c(CCNc1cc(=NCc3cn(C)cn3)[nH]cn1)cn2C c1(CCC(=O)NCCC2CCCN(C(C3CC(C)(F)C3)=O)C2)cc(F)cc(F)c1 Cc1cc(C(N2CCOC(CCCNC(=O)C3=CCC3)C2)=O)cnc1C N1(C(CCC#CC)=O)CC(NC(=O)CN2CCC(C)(O)C2)CC(F)C1 N1(C(C(C)OCCN(C)C)=O)CCCC(C)(CNC(=O)C(c2ccccc2)O)C1 C(=O)(CCP(C)(C)=O)NC(C(C)C)(C)CNC(c1cn(C)nc1OCC(F)F)=O Cn1cnc2c(N3CCC4NCCC4C3)nc(=NC(CCO)C3CC3)[nH]c12 O=C1Cc2ccc(-c3ncsc3C3(CN4CCCC45CCCNC5=O)CC3)cc2N1 Cc1nc(C=CC(=O)NC(C)C(C)(C)NC(C2CC(F)(F)C2)=O)cs1 N(C1CCc2cc(CNC(=O)C(F)(F)c3nccs3)ccc21)C(C(CC=C)C)=O C1(NC(C2C(=C)C2)=O)CN(C(=O)CCS(=O)(=O)Cc2ccccc2)CC2(CC2)C1 CCCCCCC(C)C(=O)N(C(C)CC(N1C2CSCC1C2)=O)C CC(C(C)(C)C(=O)N(C1CCOCC1)C)NC(c1ccco1)=O Cc1cc(N2CCC(C(C)NC(c3cc(=O)cc[nH]3)=O)C2)n2ncnc2n1 C1(OC)CN(C(C2(NC(c3cnc(N(C)C)s3)=O)CC(F)C2)=O)CC12CC2 C1(C(=O)NCC(=O)N(C)CC)CCCCN1C(c1c[nH]c(=NC)s1)=O C(c1ccc(O)cc1)=CC(N1CCC(c2ccccc2)(NC(C(C)C)=O)C1)=O Cc1nc(O)nc(O)c1NC(C1CC(O)CN1C(c1c(Cl)cc(Br)cc1Cl)=O)=O N1(C(CCNS(CC)(=O)=O)=O)CCC2(C1)CN(C(C1CC(F)C(=O)N1C)=O)C2 c1(C(N2CC(CC(C)NC(C3(C#C)CCCC3)=O)C2)=O)cccc(=S)n1O C1(C(N(C)CC2OCCN(C)C2)=O)CC(O)CCN1C(C1COCCO1)=O N1(Cc2c(C)n[nH]c2C)CCC(O)C(C(=O)Nc2ccc(OCC(C)C)cc2)C1 C1(CC(=O)N(C2CCN(C(C3(C(=O)OC)C=CCC3)=O)C2)C)CCC(C)(C)CC1 CC(C)(CCCCNC(=O)CCCF)NC(C1C=CCC1)=O C12(CNC(C(C)C(C)(F)F)=O)CCCC1N(C(c1ccncc1F)=O)CCC2 CC1(C)C(CO)CN1C(=O)CNC(=O)CNC(C1C(C#N)C1(C)C)=O C1(NC(CCCC=C)=O)CC(OC)C12CCN(C(c1nccn1CC)=O)CC2 C(C(F)C(=O)NC1(c2ccco2)CC1)C1N(C(=O)OC(C)(C)C)CC1 CCS(=O)(=O)CC(=O)NCC1(CNC(=O)CC=CC(C)(C)C)CC1(F)F C12(C(=O)NC(C(C)C)CCN(C(=O)C(=O)NCC(F)F)C)CC(C)(CCO1)C2 c1(CNC(CCC(C)NC(C2C3COCC23)=O)=O)cccc(O)c1F N1(C(C(C)c2cccs2)=O)CCC(NC(c2csc(C(N)=O)n2)=O)C(F)C1 N1(C(c2c(C)cns2)=O)C(C(=O)NCc2ccc(Cl)cc2)CCC12CC2 N1(C(CCC(C)NC(=O)CC2CCCSC2)=O)CCS(=N)(=O)CC1 N1(C(c2c(OCC)nc(C)cc2)=O)CCC2(CCCN2C(=O)C(C)C(F)F)CC1 N1(C(C(C)N(C)C)=O)CCN(C(C2CC3(CCC3)C2)=O)CC1c1ccccc1 N1(C(c2ccc(CC(C)C)cc2)C(=O)NCC2CC2)CC2CC(O)CC1C2 N1(C(C(c2ccn(C)n2)C)=O)CC(CNC(=O)C(O)C2CCC2)CC12CCC2 C1(C(N2CCC(C(C)NC(c3scc(OC)c3)=O)CC2)=O)CCc2c[nH]nc2C1 c1(CC(=O)NC2(C)CCN(C(C(c3scc(C)n3)C)=O)C2)ccc(Cl)cc1C C(=O)(C(O)CCC(F)(F)F)N1CCC(NC(C2CCSC2)=O)C1 c1(C(=O)NC2(CC=C)CN(c3cc(C)nc(CO)n3)C2)ccc2nc(O)oc2c1 C1(NC(=O)CCOC(F)(F)F)(CO)CN(C(c2csc(-c3nc[nH]n3)n2)=O)C1 C(=O)(C(C)(CC)CO)NCC(CC)(CC)NC(C(CCC)C)=O S(=O)(=O)(c1cccc(=NCCCCN(c2ccccc2)C)[nH]1)N(CCOC)CC c1(C(=O)NCCOCCC(=O)NCCC(Cl)Cl)cc(Cl)no1 C(=O)(C1CCCc2nc(C)[nH]c21)NCCCNC(C=C(C)c1ccccc1Cl)=O N=c1ccnc(N2CCN(C(c3oc(-c4ccccc4)nc3C3CC3)=O)CC2)[nH]1 N1(C(c2nc(C)[nH]n2)=O)CCCCC1C1(NC(=O)C(C)(C)N2CCOCC2)CC1 C1(NC(C(CC)OCC)=O)C2CC(NC(C3(N4CCCC4)CC3)=O)CC12 C1(OC)C(NC(=O)CCC2(C)CN(C(=O)COCC3CC3)C2)CC1(C)C c1(CC)cc(C(=O)NCCCC(C)NC(c2cocn2)=O)cc(C(F)(F)F)c1 C1(N(C(c2c(CC)c(C)sc2)=O)C)CN(C(C2(CCOC)CC2)=O)CCC1C C1(CNC(c2cc(CC)c(C)s2)=O)CN(C(=O)C2=CCCS2)CCC1(C)C c1(C(=O)NC2CCCN(C(CC3CC(OC)C3)=O)C2)cc(F)c(F)c(O)c1F N1(C(CCc2ccc(SC)cc2)=O)CC(=O)NC2CN(C(C3CC3C)=O)CCC12 C1(OCCNC(C=CC)=O)CCN(C(=O)Cc2nnn(C(C)(C)C)n2)C1 c1(-c2cn(C)nc2)nc(C2CC2(C)C(F)(F)F)n(CCCO)n1 Cc1cc(C(=O)NCC2(NC(=O)Cn3c(C)ccc3C)CCOC2)cnn1 O=C1CC(C(=O)NCCC2CCCN(C(c3cnnc(C4CC4)c3)=O)C2)CCN1 c1(C(=O)NC2CCC(C)N(C(=O)Cc3cnc[nH]3)C2)noc2c1CCCCC2 C1(C(=O)Nc2cc(C(=O)OC)c(C)s2)Cc2ccccc2OC1C(F)F CCC(C)(CCNC(=O)CC(=O)N(C)C)NC(=O)C(C)SC1CC1 C1(NC(c2cccc(OCC#C)c2)C2CCCCC2)CCC(=O)NC1C c1(OC)ccc2nc(C(=O)NC(C)CCNC(=O)C(N3CCSCC3)C)cn2n1 c1(C2N(C(C(=O)NN3CCCOCC3)=O)CCC2)ccc(C(F)(F)F)cc1 C1(CNC(C(=O)N(CC(=C)C)C)=O)CCCC(C(F)(F)C(=O)OC)C1 Cc1[nH]nc(Cl)c1C(=O)NC(C1CN(C(c2cc(C(C)(F)F)on2)=O)CCO1)C Cc1cc(C(=O)NCC2CN(C(=O)C(c3ccncc3C)C)CCO2)cc(N)c1 N1(C(c2c(SC)n(C)nc2)=O)CCOC(C)(CNC(c2cnns2)=O)C1 CC1(CNC(c2ccn(CC(F)F)n2)=O)CCCN1C(c1cc(C(N)=O)co1)=O CC1C(=O)NCCCN1C(=O)ON1C(C(=O)OC(C)(C)C)C(C)(C)CCC1 N1(C(=O)CCc2ccc[nH]2)CCC2CCN(C(c3ncc(Cl)cc3F)=O)C2C1 C1(C2CCOCC2)(C(=O)NCC(CNC(c2c(C)nc(C)[nH]2)=O)O)CC1(F)F C=C(C)CCC(=O)NC1CC(C)(CNC(c2cc(C)n(C)n2)=O)C1 Cc1noc(C)c1CSCCC(=O)N(C)CCOCCNC(c1ccc(F)o1)=O C1(NC(c2cc(CC)no2)=O)CN(C(=O)C(c2cnn(CC)c2)=O)CC(C)(C)C1 C1(NC(c2c(OC)nsc2)=O)CC(F)(F)CC1NC(c1c[nH]nc1C)=O Cc1cc(C#N)ccc1C(N1CC(CNC(=O)CC2CCC2C)CC(C)C1)=O Cc1ncc(NC(=O)NCCNC2CCN(C(=O)OC(C)(C)C)C2)c(Cl)c1 C1(NC(c2cc(OC)nc(C)c2)=O)CC2CCC(C1)N2C(C1(S(N)(=O)=O)CC1)=O c1(CNC2CCN(C(=O)CCc3ccco3)C2)cc(Cl)c(Cl)cc1Cl C(c1ccc(O)cc1Cl)=CC(N1CC(NC(c2ccc(Br)c(Cl)n2)=O)C(F)C1)=O C=C(C)CN=C(NCC1(C#N)CCCC1)N1CC(OC)C(O)C1 c1(NC(C2CC(NC(C3CC4(CC(C)C4)C3)=O)C2)=O)cn2ccccc2n1 C#CCC(C)(C)C(=O)N1CCN(C(=O)C(CC)OCC)C(c2ccccn2)C1 c1(C(C(=O)NCCCOCCCNC(Cc2ccc(C)o2)=O)C)ccc(Cl)nc1 c1(CC(=O)NCC(CC)N(C(=O)C(c2cccc(C)c2)C)CC)ccncc1C N1(C(C(CC)C)=O)CCCC(N(C)C(c2ncc(OC)cn2)=O)CC1 C#Cc1ccc(C(=O)NC2CC3CC2CN(C(=O)C(C)(C)CF)C3)c(C)c1 C1(CNC(Cc2cn(C)nc2)=O)CC12CCN(C(C1CC(=O)CC(=O)N1)=O)CC2 CCC(C(=O)N1CCC(CCC(=O)NC(C)C(C)O)C1)NC(N)=O c1(CN(C(C2C(C)(c3cccs3)C2)=O)CC2CCC(=O)N2)ncccc1Br c1(OCC)ccc(NC(=O)C(=O)NC2CCN(c3sc(C)cc3C)C2)cc1OC CC1CCCC(C(=O)N(CCCNC(C2CC2F)=O)C2CC2)C1 c1(N2CCCC(CNC(C(c3ccc(C)cc3)C)=O)C2)ncc([N+](=O)[O-])c(C)n1 c1(CNCC(COC)OC)c(C)nn(-c2ccc(F)cc2)c1Cl C(=O)(C1=CS(=O)(=O)c2ccccc21)NC(C(C)C)(C)CNC(=O)CCCC#N c1(CCCOC(c2csc(NC(=O)OC(C)(C)C)n2)=O)ccc2nccnc2c1 N1(C(Cn2ncc(C)c2)=O)CCC(NC(=O)CC2CC(=O)C2)C(C)(C)C1 CC(C)C(CN(C)C)C(=O)N(C1CCN(C(=O)COC2(C)CCOCC2)C1)C CC(CN(C)C)CCC(=O)N1CCCCC1C(=O)N(CCCC(O)CO)C c1(C(N2CCOCC(NC(C3(CC)COC3)=O)C2)=O)cccc2ccsc12 Cc1ccc(C(=O)NCCC(=O)N(C)CCF)o1 c1(OC)ncc(C(=O)NCC2(C)CCC(NC(C3(SC)CC3)=O)C2)cc1Cl C(N=c1[nH]c2c(c(=NCCS(=O)(=O)C(F)(F)F)[nH]1)CCC2)C1CN(C)C(=O)C1 N1(C(CSCCC(C)C)=O)CC(O)CC1CNC(=O)C(C)C(F)F C1(C)(NC(c2nc(C(C)OC)sc2)=O)CCN(S(N)(=O)=O)CC1 Cc1ncc(C(N2CC3(CCN3C(=O)COCC3CCCCO3)C2)=O)c(O)n1 c1(C(C)OC)nc(C(=O)NC2CC2CNC(=O)C(Br)=C(C)C)co1 [N-]=[N+]=NCCCC(=O)NC1C2CCN(C(C3CCCC(=O)N3)=O)CC12 c1(C(=O)NCCC2N(C(CSCC)=O)CCCC2)ccsc1S(C)(=O)=O C(=O)(CC(C)(O)SC)OC.C12C=CC(C1)NC(c1cccs1)C1CC(C1)C(=O)N2 C1(CNC(c2cnc(Cl)cn2)=O)C(C2CC2)CCN1C(C1C2CCCC12)=O c1(C(N2CC3CN(Cc4ccc5cc[nH]c5n4)CC3C2)=O)cc(F)c(Br)c(F)c1 CCC(CC)(C(=O)NC(C)C(CO)NC(c1oc(C(F)(F)F)nc1C)=O)OC C(=O)(C1=CC2CCC(C1)C2)NC(CCSC)C(=O)N1CC(F)(C#N)C1 C(C)(C(O)C(=O)NCC(C)(C)NC(=O)CSc1ccccc1Cl)SC C(=O)(C#CC1(C)CCCO1)NC1(CNC(c2ccc(C)c(Cl)c2)=O)CCOC1 C1(NC(C(CC2CC2)NC(=O)CC=C(Cl)Cl)=O)CC2(CCOC2)C1 C1(N(C(C)C)C(c2ccncc2)=O)CCC(NC(C2(C)C3COCC23)=O)CC1 Cn1cc(N)c(C(=O)NCc2ncccc2CNC(=O)Cc2ccc(F)cc2)n1 c1(SC)ccc(CCC(N2CC3CC3(CNC(c3cc(C)nn3C)=O)C2)=O)cc1 c1(CC(=O)NC(C2CCN(C(=O)COC(F)F)C2)C)nnn(C(C)(C)C)n1 C1(CNC(CN2CCC(=O)CC2)=O)C2CCC1CN(C(=O)CC(Cl)Cl)C2 C1(C(N2CCN(C(C)C(=O)O)CC2)=O)CC(=O)NC1(C)C.CC(C)C(F)C(=O)N(C)C CC1CN(C(c2cncc3[nH]ccc23)=O)CCCN1C(C1CC2C=CC1C2)=O C1(CNC(C=CC=CCC)=O)CN(C(=O)C(c2nc(C)cs2)C)CCC12CCC2 N1(C(C(C2CCOC2)OCC)=O)C2CCC1CC(NC(c1cnsc1)=O)C2 c1(C(=O)NC2C=CC(C(=O)NC(CCCC)C)C2)cc(C)[nH]c1C N1(c2c(C)cncn2)CCOC2(CCC(NC(C3CN(S(C)(=O)=O)C3)=O)CC2)C1 C1(CNC(N2CCN(C(c3nccc(N)c3Cl)C)CC2)=O)CCCC12CCC2 C12(NC(=O)Cc3cnc[nH]3)CCCC(CN(C(c3ccc4n[nH]cc4c3)=O)C1)C2 c1(N(C)C)nc(Cl)c(C(N2CCCCC2CNC(=O)C#CC2CC2)=O)s1 CON(CC1CC1)C(=O)C1(CNC(c2cc(C)oc2C)=O)CCCC1 c1(SC)sccc1C(c1nnnn1CCOCC)NC1CC2(CC2)C1 C(=O)(C1=CCCOC1)N1CCC(CC)C1C(=O)NCc1nc(O)ccc1C N1(CC(=O)NCC2CC(C)N(C(C3CN(S(C)(=O)=O)C3)=O)C2)CCCCCC1=O C1(CC(=O)NC(CCC(=C)C)C)CCCN(C(c2ccc(NC)cc2)=O)CC1 N1(C(C(c2n(C)cnc2)O)=O)CC2CCCC(NC(=O)CCS(C)=O)C2C1 c1(C(C(=O)NCC2CCOC2)N(C2C3COCC23)C)n[nH]cc1Br CCCC(C(=O)N(CCC(C)NC(=O)CNC(C1CCCCC1)=O)C)OCC C(C(C)(C)C(=O)NC12COC(CNC(=O)C=CC3CCC3)(C1)C2)N(C)C c1(OCCN(C2C(CCC)CCC2)C)ccc(OC)cc1 C=CCC(C(=O)N(CCNC(=O)C(C)COC)C(C)C)C(C)C C1(CC#C)(NC(C2CC(C)(NC(=O)C(C3CC(F)(F)C3)OC)C2)=O)CCCC1 C1(NC(C(CC)C)=O)CCCN(C(C2(C(=O)OC(C)(C)C)CCCC2)=O)C1 c1(CCCCC)ccc(NC(=S)Nc2cnc(C)cn2)cc1 c1(NC(c2ccc(CC)cn2)=O)cnc(F)cc1C C(=O)(CC1=CCN(C(C2(C(F)(F)F)CC2)=O)CC1)N1C(C(=O)NC)CC1 C1(NC(CNC(C)=O)=O)CCC2(CC1)CCN(c1nc(Cl)ncc1C(F)(F)F)C2 C(=O)(CCCC(CC)NC(=O)CC(C)(C)C#N)N1CCCC(CC)CC1 N1(C(=O)NCc2cn(CCCC(=O)OC)nn2)CCc2cnccc2C1 Cc1cc(N)c(C(N2CC(C3CN(C(=O)CN4CC5CC5C4)C3)C2)=O)cc1C c1(CSC)nn[nH]c1C(=O)NC(C)C(C)NC(=O)CSc1nncn1C(C)C C(=O)(C(O)C(F)(F)F)N1CCC(N(C(c2cnc(C)[nH]2)=O)CC2CC2)C1 C1(CS(C)(=O)=O)CN(C(C2C(Cl)(Cl)C23CC3)=O)CCN1C(c1cccc(O)n1)=O N(C1CCOc2ccc(O)cc21)C(=O)Nc1c(N(C(C)C)C)ccc(F)c1 CC(C)C(C(=O)N(C)CC1CN(C(C2CCCN2C)=O)C1)N(C)C c12ccnn1C2.C1(CC(=O)NCC2CC2NC(C2CCC2)=O)(N(C)C)CCC1 c1(-n2ccc(C)n2)ccc(C(=O)NCC2CCN(C(c3cncn3C)=O)C2)cc1 CCC(CN(C)C)CC(=O)N1CCC(NC(C2CCC(C)(C)OC2)=O)C1C c1(C(=O)NCC2(CO)CCN(C(c3ccsc3)=O)C2)csc2cncn12 N1(C(C2(C)CC(=C)C2)=O)CCC2(CC(NC(=O)COc3cccc(C)c3C)C2)C1 N1(C(c2cc(C)on2)=O)CCCC(C)C1CNC(=O)C=Cc1sccc1C c1(C(=O)NCC2CN(C(C3(CC#C)CC3)=O)CC2C)coc2c(F)c(Cl)ccc12 N1(C(C2(C)CC(=C)C2)=O)CC=CC(NC(=O)CCc2cc(C)no2)C1 C(=O)(C(CC(C)C)n1ccnc1)OCOCC(=O)c1cccs1.CO N1(C(CNC(=O)CCN2CCCCC2)=O)CCC(F)(F)C(Nc2ccc(Cl)nn2)C1 c1(N2C3CC(CNC(c4nc(C)sc4C)=O)C2CC3)nc2ccccc2o1 C1(CSCCCP(C)(C)=O)CN2CCC1CC2.N12CC(O)CC1COP(=O)(O)C2 N1(C(C=C=C(C)C)=O)CC(C)(C)OCC1CNC(C1CCc2ncnn2C1)=O N1(C(CC(CN(C)C)(C)C)=O)CCC2C(C1)CN2C(=O)C(=O)NCC(F)F C(=O)(CCC(C)NC(=O)CN(C)C)N(CCNC(C)=O)C N1(C(c2ccc(C)c(F)c2)=O)CC(NC(=O)Cc2ccnn2C)C2(CCC2)C1 CC1(C)CC(NC(=O)CCCC2CCOCC2)CN(c2ccc(C#N)nn2)C1 S(=O)(=O)(c1ccc(N2CC3CCC(C2)O3)cc1Br)N1CC(c2ccc(C)cc2)C1 CN1CCN(CCNC(C2(C3CCCN3C(=O)CCc3ccsc3)CC2)=O)CC1 c1(NCCC2CCN(C(c3c(OC)nsc3)=O)CC2)nnccc1C#N C1(OC)CCN(C(c2ccc(CNC(c3scnc3Cl)=O)cn2)=O)C(C)C1 C1(O)(CNC(C(C(C)O)NC(c2ccc(C)o2)=O)=O)CC2C=CC1C2 C(CNC(C1CCC(=O)N1C)=O)(C(C)C(C)C)NC(c1ccnc(OC)n1)=O C#CC1COCCN1C(=O)CCCCNC(c1cc2n(n1)CCO2)=O CC1CN(C(C2CC3C=CC2C3)=O)CCN(C(C2(Cl)CC2(F)F)=O)C1 c1(C(=O)NC2CC2NC(C2CCC(CCO)CC2)=O)n[nH]c2ccccc12 N1(C(c2c(C)snn2)=O)CC(NC(=O)Cc2nc(C3CC3)nn2C)C(C)C1 C(=O)(C1=C(C)CCCC1(C)C)N1CCC(NC(C(C(CC)C)O)=O)(COC)CC1 C1(OC)CCCN(C(=O)CC2CN(C(c3cc(CCO)on3)=O)CC2C)CC1 C(=O)(CCCCCN(C)C)NC(CNC(c1cnn(CCCC)c1C)=O)(C)CC c1(C(=O)NC2CCC(NC(c3c(COC)ncs3)=O)C2)cnc2[nH]c(C)nc2c1 N1(C(c2n[nH]c(C)c2Br)=O)CCCN(C(C2CCCOCC2)=O)CC1C C(N=c1ccc(Br)c(S(=O)(=O)NCC(Cc2ccoc2)CO)[nH]1)C1(C)CCO1 C1(CNC(CC2CC(=C)C2)=O)C2CCC(C2)N1C(=O)CNc1nccs1 c1(N2C(c3ccc(OC)cc3)CSCC2)cncc2nnnn12 c1(C(=O)OC)nc(Br)ccc1NC(C1(O)CCN(Cc2c(C)cccc2Br)C1)=O Cc1ccccc1C(CN(c1nc(CC(F)(F)F)ns1)C)Nc1ccccc1 C1(CN(c2ccc(C(=O)OC)cn2)C)C2CCC1CN(C(=O)CN1CCCC1C)C2 c1(CCNC(N(C)Cc2nc(CC)on2)=O)cnc2ncccn12 C(=O)(C(CC(C)(C)C)OCC(CCOC(C1(C(CC)(F)F)CC1)=O)OC)NCC C(=O)(C1=CCOCC1)N1C(C)CC(NC(C(C(C)C)NC(C)=O)=O)C1 n1(CC)ncnc1C(=O)NC1CCCC1NC(=O)CCc1ccccn1 C(=O)(C(O)C(C)(C)CC)N(CC(=O)N(C)Cc1cncs1)CC#C c1(C(=O)OCC)cn2c(C(=O)NCCN(C3CCS(=O)(=O)C3)C(=O)OC)cnc2s1 N1(C(Cc2cc(C)on2)=O)CCC(C2CC2)C1C(=O)NOCC(O)C(C)C N1(C(CCN(CCCCC)C)=O)CC2(C)CN(C(C3(C)CC3Br)=O)CC2(C)C1 C1(C2CCC2)(CNC(C2CCCN(Cc3ccccc3)C2)=O)CC1 c1(CN(S(=O)(=O)CC2(C#N)CC2)CCOC)ccc(F)cc1Cl Cn1nc(C(N2CC(C(O)C(=O)NCc3nc(=O)o[nH]3)C2)=O)cc1O c1(CCCC(=O)NCC2CC2CNC(c2ccccn2)=O)c(F)cccc1F Cc1nc(C)n(CCCC(=O)NCC2CCC(NC(=O)C(F)(F)CO)CC2)n1 C1(CNC(C=CC(C)C)=O)CC2(CO1)CN(C(=O)C(C)C(F)F)C2 C1(CCC)(NC(=O)CCC(C)N(C)C)CCN(C(C2CCCS2)=O)CC1 CCCCCCCCC(C)C(=O)N(CCOCCO)CC.C1(=O)C(C)(C(C)C)N1 c1(C(=O)NC2(CNC(c3ccc(O)c(Cl)n3)=O)CCCC2)ccc2c(c1)CCO2 N1(C(C(CCN(C)C)O)=O)CC2CC1CN(C(=O)CN(CC(C)(C)C)C)C2 c1(CCS(=O)(=O)N(CC(N2CCC(C(C)N)C2)=O)C)ccc(O)cc1 c1(-n2ccc(CNC(=O)C(=O)NCC3(OSCC4CC4)CC3)n2)ccccc1Cl N1(C(C(=O)NCc2nnc(COC)s2)=O)CC2NC(C1)c1ccccc12 C(N=c1cc(C(F)(F)F)nc[nH]1)C1CC(NC(CC(C)c2cccnc2)=O)C1 C1(NC(=O)CCOCC(F)(F)F)CN(c2cc(O)nc(O)n2)C2CCCCC12 c1(OC)ccc2occ(C(=O)NC3CN(C(=O)CC4CCOC4)CC34CC4)c2c1 C12(C(N(C3CN(C(C4CCc5ccnn5C4)=O)C3)C)=O)CCC(F)(CC1)CC2 Cc1ccc(Br)c(C(C(=O)Nc2ccc(F)cc2C)N(CCCC2(C)CC2)C)c1 N1(C(c2cc(C(=O)OC)c(F)cc2)=O)CCC2(C(=O)O)CCCC12 CC1(C)CN(C(=O)CC23CCC2CN(C(c2cc(F)cnc2O)=O)C3)CC1CO c1(C(N2CCC(O)(C(C)NC(C(F)=CCC)=O)CC2)=O)c(C)cc(C)cc1N c1(N2CCC(C)(CC)C2)ccc(S(=O)(=O)NCC#Cc2ccc(F)cc2)cn1 C(=O)(C(CCC)C(=O)OC)N1CC(C2(NC(C(CCCC)N(C)C)=O)CC2)C1 N1(C(COC(CC)(C)C)=O)CC(C)CCC1CNC(=O)COc1ncccn1 C1(C2CC2)(C(=O)Nc2cc(C(N)=O)[nH]n2)CNC1 c1(C(C(=O)NCC2(C(C)NC(=O)C(C)(C)CO)CC2)=O)cc(Cl)cc(Cl)c1 N1(C(CNC(=O)OCC=C)=O)CC2(CCC2)CC1C(=O)NOCCC(=C)C C(C(O)CC(=O)NC1CC1)NC(=O)CC1CCCC12CC2.C12(CCCC1)C(=O)N2 N1(C(c2c(C)nn(CCO)c2)=O)CCN(C(C2CC2C)=O)CC1c1ccncc1 c1(C(N2CCN(C(c3c(OC)nc(C)cc3)=O)CC2)=O)cnn2c1CN(C)CC2 C1(CNC(C(=O)NCC)=O)CCN(C(C23CC(CO2)C3)=O)C1c1ccccc1 c1(-n2cc(CC3CCN(C(C4CC(C)SCC4)=O)C3)nn2)cccc(Cl)c1F c1(CSC)cc(C(N2CCC(CNC(=O)C(C)C(F)F)CC2)=O)sc1C C(=O)(C#CC1CCCOC1)N(C1CCCC1NC(c1ncccc1N(C)C)=O)C c1(C(N2CC3C(CNC(c4c[nH]c(=NC)s4)=O)(C3)C2)=O)c[nH]c2ccc(Cl)cc12 C1(NC(C(=O)NCC(CC(=O)OC)C2CCC2)=O)CCN(C)C(=O)C1 C1(F)(CNC(C(CSC)C)=O)CC2CCC(C1)N2C(=O)CNC(N)=O N1(C(CCOCCC)=O)CCC(NC(=O)CN(C)C)CC1c1ccccc1 c1(OC)ccc(CC(N2CC(O)(C(C)NC(=O)C(C)C3CC3)C2)=O)cc1F O=c1cc(CNCc2csc(-c3cscn3)n2)[nH]c2ccccc12 c1(NC(=O)CC2CN(C(c3ccc(CO)s3)=O)CCO2)cnn2cccnc12 c1(C(=O)NC2CCC(N(C(=O)CCc3cnn[nH]3)C)C2)nc(Cl)c(=O)[nH]c1N c1(CCC)ccccc1CCn1cc(CC(=O)N(CCCOC)C)nn1 c1(C(=O)NC2CN(C(C=C(C)C(C)(C)C)=O)CC(O)C2)cnc2n(c1=O)CCS2 N1(C(c2c(SC)scc2)=O)CCC2(CC1)CC2CNC(C1CCNC1=O)=O CCC(C)C(O)C(C)C(=O)NC(C1CCCN1C(c1cc(C(F)F)[nH]n1)=O)C C12CC(CC1O)CNC(=O)C1(CC1)CC(=O)N2.N1(C(=O)OC)CC=CC1CF c1(C(=O)NCC2CN(C(Cc3ccc(C)nc3)=O)C(C)C2)cnc2sccn12 C(=O)(C(CC(F)F)NC(=O)CC1CCC(=O)NC1)Nc1c(OC)nn(C)c1 C(=O)(CN=c1cc[nH]cc1)N1CCCC(O)(CNC(c2n[nH]cc2F)=O)C1 CCC(C)CCC(=O)NCC(O)CNC(c1c(-c2ccccc2F)noc1C)=O C1(CC=C)(NC(=O)C(F)(F)CN(C)C)CCN(C(c2ccsc2Cl)=O)C1 N1(CC(=O)NCC(C)CN(C)C(C2CC(C(F)F)C2)=O)CSCCSC1 Cc1ccc(C(C)C)cc1.C1(=O)C(C(C)C)SCCC(=O)N(C(C)C)CCN1C Cn1cccc1C=CC(=O)NC1(CNC(C2CCCCC2)=O)CCOC1 CC12CN(C(=O)CC3(O)CCOC3)C(C(=O)NC3CCC3c3ccccc3)(C1)C2 C(=O)(C(C)(C)CC(=O)NCc1ccnc(C(=O)NC(C)(C)C)c1)OCC C(=O)(C1CCCc2sc(C)nc21)NCC(CCOC)NC(=O)Cc1ccccc1 C1(CC(=O)NCC2CCC(=O)C2)CC(F)CN1C(c1ccoc1)=O n1(CC(N2CCN(C(C3C(C)(C(C)C)C3)=O)C(C)C2)=O)nc2n(c1=O)CCCC2 C(C#Cc1cccnc1)NC(CCC1CCCN(C(c2cnc(OC)s2)=O)C1)=O CC1CC(COC(=O)CCCSc2ccc(N)cc2)CC(C)C1 C1(C(=O)NCCC(C#C)(C)C)C2CC3C(C2NC(c2ncncc2N)=O)C13 c1(C(N(C(CCNC(C2C(C(C)C)CCC2)=O)C)C)=O)cn2cc[nH]c(=O)c2n1 N1(C(c2n(CC)ncc2)=O)CCCN(C(=O)C(F)(F)C2(O)CCCC2)CC1CO C(C(C)(C)CC(=O)N1CC2C(NC(C3CCCN3C)=O)C2C1)N(C)C C(CC(=O)NCCN(CCC(N)=O)C(=O)C(C)OC1CCCC1)C(C)C C=CC(C)(C)C(=O)NCC(O)CCNC(c1cc(-c2ccc(C)cc2)n(C)n1)=O c1(N(CC(=O)NCCN(C(C2CC2(F)Cl)=O)CC)C)ccnc(Cl)n1 C(C(O)C(F)(F)F)NC(C1CCN(C(Cn2c(C)ncc2)=O)C1)=O c1(OCC(=O)NCC(C)(N(C(=O)C(=O)NC2CC2)C)C2CC2)ccc(F)cc1 Cc1c(C)c(C)c(C(=O)NCC(F)CNC(c2cnc3n2CCC3)=O)c(C)c1C c1(OC)cccc(C(N2CC(NC(c3ccc(C(N)=O)cc3)=O)C3CC23)=O)c1N C1(C)(CC(=O)NC(C2(CNC(=O)CC(C)c3ccco3)CC2)C)CCCO1 Cn1ccnc1CCC(=O)NCCCNC(C1CCC1(F)F)=O C(CN=c1ccn2ccnc2[nH]1)(C1CCCCC1)NC(c1cc(C)sc1C)=O Cc1ccc(S(=O)(=O)N2CCN(C(C3CCC(F)(F)C3)=O)CC2C#N)cc1C Cc1cc(C(=O)NC2(C(N3CCCC3CF)=O)CCC2)nc(O)c1 C1(NC(C2N(CCC)CCC2)=O)(CO)CCCN(C(=O)C(C)(C)O)C1 C1(CC(=O)NC(CNC(CSCC)=O)C(C)(C)C)CCc2ccccc2N1 Cc1ccc(C(N2CCCCC2CCCNC(C2(C)CC=CCO2)=O)=O)c(C)c1 NS(=O)(=O)c1cc(C(=O)NC(=O)CCc2ccc(O)c(O)c2)ccc1Cl c1(SCC)cccc(NC(C2CCN(C(=O)C(F)(F)CC3CC3)CCCO2)=O)c1C c1(CN(C=O)Cc2c(C)cc(C)s2)cc(Br)ccc1Br C1(NC(c2c(N)cc(Cl)cc2)=O)CC2CCC(C1)N2C(c1occc1F)=O S(=O)(=O)(c1ccc(C(C)(C)C)cc1)N1CC(NC(CCCCCCC)=O)(CO)C1 C(N=C(NC(C1(CO)CCCC1)C)NC1CCC1)C1CCN(OCC)C1 C1(NC(C=C(CC)CC)=O)CC2CC(NC(c3cc(OC)ccc3C)=O)C1C2 Cn1nc(Br)cc1C(=O)NC1(CNC(C2CCCCC2O)=O)CCCC1 N1(c2ccc(CC(C)C)s2)CC(CO)OC(CO)C1 N1(C(C2CCCC(=O)C2)=O)CC(=O)NCC1C(=O)NCc1ccc(F)cc1O C1(CCNC(CCC2CC(OC)C2)=O)CN(C(c2ccnn2CC#N)=O)CC1C c1(OC)ccc(C(=O)NC2CC(NC(C3CCCN(C)C3)=O)C2)cc1OC(F)F N1(CC2CN(C(S(=O)(=O)C3CC3)C(=O)OC)CC2CO)CCC(O)(CO)CC1 C1(CC(N2C(CNC(C(c3cccnc3)OC)=O)CCC2)=O)CCCC1C1CC1 c12nc(-c3c[nH]c(C4CCCO4)c3)n(n1)C2.N1(Cc2sccc2)CCOCC1 N1(C(C(C)(N(C)C=O)C2CC2)=O)CCOC(C(N)=O)C1.c1(C2CC2)csc(Cl)n1 C1(CC(=O)NC2CC(CC(=O)NCCCOCCO)C2)CCCCC1 Cc1ccncc1CC(=O)NC(CCF)C(=O)NCC(C)CCO CC(C(=O)N(CCCN)C(C)(C)C)C1CCNC1 c1(C(=O)Nc2nccc(-c3ccc(C(C)(C)O)cc3)c2)cc(I)ccc1[N+](=O)[O-] C(=O)(C1=NOC2(CCC2)C1)NCC(C)CN(C)C(C1CCN(C)C(=O)C1)=O c1(CCC)ccc(N)c(C(=O)NC2CC(F)CN(C(=O)CSC(F)F)C2)c1 C1(C2C(c3n(C)cnn3)CC2)(NC(=O)CC#N)CCN(C(=O)C2=CCCOC2)CC1 C1(OC)CCCN(C(=O)C(c2ccccc2)NC(c2cc(C)cs2)=O)CC1 C(=O)(C(O)CNC(=O)C(Cc1cc[nH]n1)NC(c1ncccn1)=O)NC C1(NC(c2c(C)n(C)cc2)=O)CCC2(CC1)CN(C(=O)CCC1(C)CC1)CCO2 c1(C(=O)NCc2c(C(=O)NCC3C(OC)CCC3)scc2)cccc(C)n1 c1(C(=O)NC(C2CCCN(C(c3c(C)nco3)=O)C2)C)cc2c(O)cccc2[nH]1 c1(C(N2CCC(NC(CNC(C(CC)C)=O)=O)C2)=O)ccc(NS(C)(=O)=O)cc1 CCCCCCC(C)C(=O)NC(C)CNC(c1cnc2c(c1)CCC2)=O c1(OC)cc(C(=O)NCC(C)NC(=O)COCC(F)(F)F)cc([N+](=O)[O-])c1Cl C1(O)(CNC(=O)C(F)=C2CCC2)CC(C(=O)NC2(C3CCCCO3)CC2)C1 CNS(=O)(=O)N1CCC(C(=O)NC23CC2CN(C(=O)CS(N)(=O)=O)C3)CC1 C(CC(C(C)C)NC(C1(F)CCOC1C)=O)NC(C1C(CC)OCC1)=O N1(C(c2c(C)csc2)=O)CCC(O)(CNC(c2ccccc2CO)=O)C1 C1(C(=O)NCC(CC)NC(=O)Cc2ccc(Br)s2)C2CC3C(C2=O)C13 c1(C(CC(=O)NC(C2(CNC(=O)C3=CCSC3)CC2)C)C)c[nH]c2ccccc12 C(=O)(CCC(F)(F)Cn1cc(C2(F)COC2)nn1)N(C)CCc1ccc(F)cc1 CC1=C(C)CC(C(=O)NC2CC(F)(CNC(c3c(C)ccnc3O)=O)C2)CC1 N1(CCC#C)CCC(C(=O)NCC2(F)CC(NC(=O)CCC=C(C)C)C2)CC1 N1(C(C(C)OCC#C)=O)CC2CC(C(N3CC(c4cc[nH]n4)C3)=O)(C2)C1 c1(CCC(=O)NC2CC(CCn3cc(CCCSCC)nn3)C2)ccccc1Cl C(=O)(CCCC(=O)NCCCOCCCCNC(=O)CC1CC1C1CC1)NCC c1(CC(N2CC(C)(NC(Cn3cc(C(=O)OC)nn3)=O)C2)=O)c(Br)cnn1C C1(NC(=O)Cn2cnnn2)(CO)CCCN(C(=O)CCc2cccnc2F)C1 N1(C(=O)CCOCC(F)F)CCN(C(c2cc(Cl)ncc2O)=O)C(CF)C1 C(=O)(C1CCCc2nn[nH]c21)N1CC(C)(NC(=O)COC2CCC2)C1 c1(C(N(CC(C)NC(C(CCC)(C)CC)=O)C)=O)nc2c(Br)cccn2c1N Cc1cccc(C(N2CCC(C)(CNC(=O)CCc3cccc(O)n3)C2)=O)c1O CCC1=C(C(=O)NC2CC(C)CN(C(c3ccc(F)cn3)=O)C2)CCCO1 Cc1c(C(N2CCOCC2CNC(C2CCCN2C)=O)=O)cc(N)cc1O CC(C)(CF)C(=O)N1CCC(C(C)(C)C)(CNC(=O)CCC2CCCOC2)C1 C1(C(N2C(CN(C(c3cnn(CC)c3)=O)CC)CCC2)=O)C2(CCC2)C12CCC2 c1(CC(=O)NC2C(NC(C=CC)=O)CCCCC2)ccccc1S(C)=O C1(C(N(C2CCN(C(C3C=CCC3)=O)CC2)CCC)=O)CCc2nccn2C1 C1(C(N2CC=C(CNC(c3c(OC)cccn3)=O)CC2)=O)Cc2ccccc2S1 C1(C2CCCN(C(=O)CCc3ccccc3F)C2)(NC(C2CNC(=O)N2)=O)CC1 N1(C(c2cc(C(C)=O)sc2)=O)CC2C(CNC(C3CC4CCC3O4)=O)C2C1 C1(C(N(CCCNC(C2CC(O)(C(F)F)C2)=O)CC)=O)CCC(C2CC2)C1 C(=O)(CCC(CF)CF)N1CCC(C)(C)C1C(=O)NCCOCC1CCC1 C1(NC(C(C(C)(C)C)O)=O)COC2CN(C(c3cc(C(F)F)cc(Cl)c3)=O)CC12 c1(C(=O)NC(C2CC(NC(c3nc(C)oc3)=O)C2)C)cnc2n1CCCC2 C(C)(CCC(F)(F)F)NC(COC(CNC(COCCOC)=O)(C)C)=O c1(OC)cc(Br)cc(NC(C2CCCN(C(c3ccsn3)=O)CC2)=O)n1 C1(N(C(C(C(C)C)F)=O)C)CCCN(C(C2CC2c2cnn(C)c2)=O)CC1 C(=O)(C(C(=O)N1CC(NC(c2cccnc2-n2cccn2)=O)C(O)C1)OC)OC N1(C(COCCCCC)=O)CCC(N(C(=O)CCn2ccc(C)n2)CC)C1C c1(CC(=O)NCCC(CNC(CC)=O)O)cccnc1OC C(=O)(CC(C)C(F)(F)C(F)(F)F)NC(CC)(CNC(c1c(C)ncn1O)=O)CC N1(C(C=C(C)C2CC2)=O)CC2CCC(CNC(c3nnc(C)o3)=O)C2C1 c1(C(N2CCC(C)(NC(CC3CCC(C)(C)C3)=O)C2)=O)cncc2ncccc12 Cc1ccc(C=CC(N2CCCC2C(=O)N(c2cccc(Cl)c2)C)=O)o1 C1(CCC(=O)NC(CC=C)CNC(C2(c3ccn(C)n3)CC2)=O)CCN(C)CC1 C(C(CCC)C(=O)N1CCCC(O)(CC(N)=O)C1)NC(C(C=C)OC)=O n1(C(C(=O)NC(CCC)C)C)cc(-c2ccccc2)nn1 C1(C(=O)NCCN(C(=O)C=CBr)CC)Cc2ccc(F)cc2O1 C1(C(=O)NCCN(C(=O)C(F)CC2CCCCC2)C2CC2)CCc2n[nH]cc2C1 c1(C(N2CCCC(N(C(C3ON=C(C)C3)=O)C)CC2)=O)cccc2c1cnn2C c1(C(N(CC(CN(C(c2cc(C)nnc2)=O)C)O)C)=O)nc2sccn2c1C C1(OCC)CN(C(=O)CC2CCC(=O)CC2)CC1CNC(=O)CCC1CC1(F)F Cc1ccc(NC(=O)C(C)N(C(C23CSCC2C3)=O)C(C)C)c(O)n1 N1(C(CCC(C)(F)F)=O)CCN(C(=O)C(F)C2CCCC2)C2CCCC2(C)C1 C1(C(=O)NCC(CCC)O)CN(C(=O)C(C)(C)C2CC2)CC12CC2 N1(C(C(C(C)C)NC(C)=O)=O)CCC2CN(C(=O)CC(C(F)(F)F)N(C)CC)C2C1 N(C1CCc2c(Cl)cc(Cl)cc21)C(c1ccc2scc(Br)c2c1)=O N1(CC(=O)OCC2COc3ccccc3O2)CCC2(C1)OCC1CC21 c1(CN2C3C(C(=O)Nc4nnccc4C(F)(F)F)C(C3)C2)c(F)ccc(Cl)c1Cl CC(C)C(C)C(CNC(=O)CCn1ccc(O)nc1=O)NC(c1ccsn1)=O c1(-c2ccc(C3CC(CC)OCC3)cc2)ccc(S(=O)(=O)N2CCCCC2)cc1 N1(C(C(C(C)C)F)=O)CCN(C(=O)CCN2CCN(C(C)C)CC2)C(C(F)F)C1 N1(C(C2CC23CCOC3)C(=O)N(C2(C(=O)OCC)CC2)CC=C)CCC(C)(F)CC1 N1(C(c2nncc(C)c2)=O)CCC2(CCC2)C(NC(c2ccc(F)c(Cl)n2)=O)C1 CCS(=O)(=O)CC(=O)N(CC(=O)NC1CN(C(C)=O)C1)CCOC c1(NC(C=CCN(C)C(C2CC2(F)Cl)=O)=O)ccc(Cl)c(O)c1 C(C(O)C(=O)NC1(CN(C)C(C2CCCC2c2nncn2C)=O)CC1)OC CCC(CC(=O)NCC1C(C)CCN1C(c1ccncc1Cl)=O)CC(F)(F)F c1(C(=O)Nc2ccccc2-n2ccnc2)cc2scc(Cl)c2[nH]1 c1(NC2CC(NC3N(C(C(C)OCC=C)=O)CC3)C2)cc(CC)nc(C)n1 C(c1cccc(C)c1)=CC(=O)NC(COCC)C(=O)NCCC(C)N(C)C N1(C(C(CC#C)C)=O)CC(CNC(C2(C3CC3)CC2)=O)C2(CC2)C1 c1(C(N2CCC(OCCNC(C3C(C)CCS3)=O)C2)=O)cc2n(n1)CCCO2 c1(CNC(c2n(CC)nnc2)=O)ccc(C(=O)NCCC2CCCC2(C)C)cc1 Cn1cc(Cl)c(C(=O)NC2CN(C(=O)COCP(C)(C)=O)CC2O)n1 CCC(C)(C(=O)NC1CN(C(=O)COCc2ccnn2C)CC1O)C(F)F S(=O)(=O)(c1ccc2sc(Cl)cc2c1)OC.c1(N2CC2=O)cc(C)ccc1C#N N1(C(C(C)N2CCC2)=O)CCN(C(C2CCSCC2)=O)CC1CC(C)(C)C [N-]=[N+]=NC1CC(C(=O)NCCCC2(O)CC2)N(C(C2(O)CCCCC2)=O)C1 N1(C(c2c(C)ccc(F)c2)=O)CCOC2(CCN(S(=O)(=O)C(F)(F)F)CC2)C1 C1(N(C(=O)CC2CCCOC2)C)CCN(C(=O)CNS(=O)(=O)C2CC2)CC1 c1(-c2c(C)csc2)cnc(F)c(C(=O)Nc2ccnc(F)c2C)c1 CCC(CC)CC(F)C(=O)NC1(C(=O)NC2(C)CCCC2(C)C)CCSC1 c1(OC)ccc(Cl)c(C(N2CC(NC(=O)CNc3ccccn3)C(C)(C)C2)=O)c1 O=C(CCCc1ncco1)NC1(CCNC(C2(F)CC=CC2)=O)CCCC1 c1(C(N2CC(NC(c3c(C)nn[nH]3)=O)C2)=O)cnn2c(-c3cccs3)ccnc12 c1(C(=O)NCC2CCC(NC(c3nc(C(C)C)oc3)=O)C2)nnc(S)n1C C1(NC(C(C)CC2CC2)=O)CCCCN(C(c2cnn(C)c2Cl)=O)C1 C(=O)(CCCCC(F)(F)F)NC1C(CNC(C2C(C)(C)CCCO2)=O)CCC1 CCN=C(NCCC(N1CCOCC1)C)NCC1CCOC1(C)C Cc1cc(CCC(=O)N(C(C)CNC(c2ccc(Cl)[nH]2)=O)C)ccc1Cl c1(C(=O)NCC2(CNC(C(C)SC(F)(F)F)=O)CCC2)c[nH]c2cnccc12 c1(C(C(=O)NCC(C2CCOC2)OC)OC(=O)N(C)C)cc(F)ccc1F C1(NC(C(=O)NC(C2(O)CC2)C)=O)CC12CCCc1ccccc12 N1(C(C#C)C)CCN(C(=O)CC2CCC(NC(c3cc(CCC)[nH]n3)=O)C2)CC1 C1(c2c(OC)cccc2)CCC(C)CN1C(=O)CSc1ccccc1C c1(OC)cc(Cl)c([N+](=O)[O-])cc1C(=O)Nc1cccc(C=CC(F)(F)F)n1 n12cc(nn1)CNC(=O)C21CC1.C1(C(=O)NC(C2(CO)CC2)C)CCOC1C C1(C(=O)NCCCNC(CCc2n(C)cnc2)=O)CCCCS1(=O)=O c1(CC(=O)NC2C(NC(C(CC=CC)C)=O)CCCC2)ccc(C#N)nc1 O(N=C1CCCCCC1)CC(N1CC(C)C(NC(c2cc(C(N)=O)c[nH]2)=O)CC1)=O N1(C(C)=O)CCC(C)C2(CCCCC2)C1.S(=O)(=O)(c1cccnc1)N1CCCCC1 c1(CC(=O)N(C(Cc2ccccc2)C(=O)OC)CC)cccc2c1OCCO2 c1(C(=O)NCC2CN(C(c3ccc(Br)o3)=O)C3CC23)cc2sccc2cn1 c1(CC)nc(C)c(CNC2CCN(N(C(=O)C(C3CC3)OC)C)C2)o1 c1(C(N2CCC(C(C)NC(c3sc(F)cc3Cl)=O)C2)=O)nn(C)c2ccccc12 C(=O)(CC(C)CC(F)(F)F)N(C(CNC(c1cc(C)c(F)cc1F)=O)C1CC1)C c1(C(=O)NC(COC(C)C)C(=O)N2CC(C(N)=O)C2)ccncc1N C1(COCC(=O)NC2CC2CNC(CC2(C(=O)OC)CC2)=O)CCCO1 N1(CC(=O)Nc2c(C)ccc(C)c2)C2CCC1CN(C(=O)C(C)CC(C)C)C2 Cc1ccn2ncc(C(=O)NC3CCC(NC(C4CN(C)CC4C)=O)CC3)c2n1 CC1(C(N2CCOCC2)=O)CN(C(C2CCS2(=O)=O)=O)C1 C1(CN(CCC(=C)C)Cc2ccco2)CCCCC1 N1(C(c2c(CC)nc(C)o2)=O)CCC(C2CCN(C(C3(C)CCC3)=O)CC2)CC1 N1(C(C(C(=O)OC)OC)=O)CC2(CCCC2NC(=O)CCC=C(C)C)C1 N1(C(c2cc(COC)no2)=O)CC(NC(=O)C(C)NC(C)=O)C(C)C1 Cc1cc(C(N2CC(F)(F)CC2C(=O)Nc2cncc(C#N)c2)=O)cc(C)n1 Cn1nc(C(=O)NC2CCCCN(C(c3n[nH]c(O)n3)=O)C2)c2c1CCC2 C1(NC(C2C(C)CCCC2)=O)C2CC3C1C3C2C(=O)NC(C1CCCC1)C c1(C(=O)NC2(CNC(c3ccc(OC)s3)=O)CCCC2)cccn(C)c1=O CCCCC(C)C(=O)N(C)Cc1ccc(CNC(C2CC2C2CC2)=O)cc1 CCC(C(=O)NC1CC(NC(c2cc(=O)c(OC)c[nH]2)=O)C1)C(C)(C)CC C(=O)(C(F)(F)C(F)(F)C(F)F)NCC(C)NC(=O)CNC(=O)C1CC1 c1(CC)nc(Cl)nc(N2CCC(C3(NC(=O)C=CC4CCC4)CC3)C2)c1Cl C(C)(CS(C)=O)NC(CN(C(=O)CC1CC1CC)CC#C)=O C(=O)(CC1=CCOCC1)NCC1CN(C(c2ccc(C(=O)OC)s2)=O)C(C)CC1 C12(C(N3CC(C)(CCC(=O)NCCN(C)CCO)C3)=O)C(=O)C3CC1C2C3 CCC(CC(=O)N(C1CC(NC(c2sccc2OC)=O)C1)C)CC(F)(F)F c1(CC(=O)NCCN(CCC)C(c2cnn(CC)c2)=O)csc2cc(C)sc12 c1(C(=O)NC2CCC(CC(=O)NC(c3cnccn3)C)C2)ccnnc1O c1(C(N2CCC(CC=C)(NC(C3CC(Cl)(Cl)C3)=O)C2)=O)cnn2c1CCCC2 C1(CC(=O)NC)CN(C(C2CCOC2C2CC2)=O)CCN1C(c1ccc(Br)o1)=O N1(C(C2C(OC)(OC)CC2)=O)CC2CCCC1(CNC(=O)C=C1CCOCC1)C2 C(=O)(C#CC1CCCO1)NCC1(CNC(C2(C#N)CCC2)=O)CCC1 c1(C(N2CCCCC2)CNC(=O)NCCC(=O)Nc2ccoc2)ccccc1 C(=O)(C(C(=O)NCC1(NC(=O)C(C)Oc2ccc(F)cc2)CCC1)OC)OC c1(C(N2C(C(C)NC(c3cc(CC)on3)=O)CCCC2)=O)nccc2[nH]ccc12 c1(C(N(CCCNC(CC2(C=C)CC2)=O)C)=O)cc(F)c(F)c(F)c1N N1(C(C=C(C)C2CCCCC2)=O)CC2(CCCC2NC(=O)C=C2CCOCC2)C1 C1(CCNC(C(CNC(=O)CCC2CCCO2)OC)=O)CCCC1(C)C c1(CNC(C(n2c(C)ncc2)C)=O)cccc(C(N2CCCC(C(F)F)C2)=O)n1 C1(C(=O)N)CC2(CC2)CO1.C1(C(C(=O)CCCC2(CN)CCC2)=O)CC(F)(F)CS1 N1(S(=O)(=O)CC2CCC2)CC2CCC(C1)N(CC(F)(F)F)C2 c1(C(N(C2CCN(C(c3ccccc3F)=O)CC2)CCO)=O)cc(Br)ccc1F C(=O)(C(C(C)OC)N(C)C)N1CC(C(=O)NC2(COC)CC2(C)C)(CC)C1 C(S(C)(=O)=O)C1(N(CCCN(C(=O)CC2(C(F)(F)F)CC2)C)C(C2(C)CC2)=O)CC1 c1(C(=O)NC23CCN(C(=O)C4=COCCC4)CC2C3)nccc2ncccc12 C1(NC(C(C2CC2)OC)=O)CCC(NC(=O)CCN2CCCCC2)CC1 C1(NC(c2cc(CC)on2)=O)CCCC12CCN(C(c1ccc(F)cc1O)=O)C2 c1(C(N2CC3CC2CN3C(c2ccc3nc[nH]c3n2)=O)=O)ccnc2cc[nH]c12 c1(C(N2CCC(=C)CC2C(=O)NCC2(C#N)CCCC2)=O)nccc2[nH]ccc12 N1(C(CC2ON=C(C)C2)=O)CCCN(C(=O)CCC2CCC(=O)N2)CCC1 Nc1ccnc2c(C(N3C4CCC3CN(C(C3CC3Cl)=O)C4)=O)cnn12 Cc1ccc(C=CC(=O)NC2CC(=CC(=O)N(C)C3CC3)C2)cc1 C(CN=c1ccnc(NCc2c(O)cccc2Cl)[nH]1)OCC(C)C C(c1ccccc1[N+](=O)[O-])=CC(=O)NC(C(C)C)(C)CNC(C1(O)CC1(C)C)=O Cc1[nH]c(C#N)cc1C(=O)NC1(CF)CN(C(C2CCCC2(F)F)=O)C1 C=CC(C)(CC)C(=O)NCC(C(C)(C)C)NC(c1ccc(=O)n(CC(C)O)c1)=O C1(NC)CCCCCC1CNc1cc(N(C)Cc2cccc(C)c2)nc(C(C)C)n1 C(=O)(C1(C)Cc2cccc(Cl)c21)N1CCCC(C)(NC(c2cc(CC)on2)=O)C1 C1(C(N2CC3(CC(NC(CCC(=C)C)=O)C3)C2)=O)CC2(CCCCC2)S1(=O)=O S(=O)(=O)(c1cccnc1NCc1cc(Cl)ccc1F)NC(C)Cn1cccn1 N1(C(CC2C(=O)NCC2)=O)CC2CC1CN2C(c1cccnn1)=O C1(C(N2C(CCCNC(C3N(S(C)(=O)=O)CCC3)=O)CCC2)=O)CCC2CC2C1 c1(CNCC(C)CC2CCCCC2)nn(C(C)C)cc1Cl C1(C(=O)NCCCOCC=C)CC(C)(C)CCN1C(c1cscn1)=O C(=O)(C1CCCc2ncnn21)NC1CC2CN(C(c3c(CC)nn(C)c3)=O)CC21 N1(C(C(C)NC(N)=O)=O)CCOC(CN(C)C(C2CC(C)(C)C2)=O)C1 C12(C(=O)NC3C(C)CN(C(C45CCC(C)(CO4)C5)=O)C3)CC(C)(C1)OC21CCC1 c1(C(=O)Nc2nc(C)c(C(=O)O)s2)nccc2ncncc12 c1(NCC(CCCC)NC(=O)C(C)CC2CCC2)nnc(C)c(C)c1C#N N1(C(c2cnc(OCC)s2)=O)CCN(C2CC2)CC(NC(=O)CCOCOC)C1 C1(C)(COC)CCCN(C(c2cnc(-n3cncn3)nc2)C(=O)NC(C)(C)C)C1 Cc1[nH][nH]c(=NC(=O)C2c3ccccc3CN2C(c2cnco2)=O)c1C c1(CNC2CCCC(C(N(C)Cc3ccncc3)=O)C2)c(Cl)cc(Br)cc1Cl c1(OCC(=O)NC2CCCC2NC(C2CCCOC2)=O)ccc2c(c1)CCC2=O c1(C(=O)NC2CC(CNC(C(C(C)O)C)=O)C2)cnc(O)nc1O c1(OC)ccc(Cl)c(C(=O)NC23CC(NC(=O)C(CSC)OC)(C2)C3)n1 C(N=c1[nH]nc(C(F)F)s1)C1C(C(F)(F)F)CN(C(c2c(CC)ocn2)=O)C1 c1(OC)ccc(C(=O)NC2CN(C(=O)CN3CCC3CO)CC2C)c(F)c1F N1(C(c2cnc(N(C)C)nc2)C(=O)NCC=C)CCOCC12CNC(=O)OC2 C1(CNC(=O)CCNC(=O)C2CC2)CC(C(=O)Nc2ccccn2)C12CCC2 C#CCC(C(=O)NC(c1ccccc1)CNC(=O)COCC1(F)CC1)C1CC1.OC C(C)(CCCCNC(=O)CC(C)NC(N)=O)NC(CCc1cc(C)[nH]n1)=O C1(CNC(c2csc(-c3nc[nH]n3)n2)=O)CC2(CO1)CN(C(C1C=CCC1)=O)C2 CC(C)C(C(=O)NCC1C2CN(C(C3CCCCO3)=O)CC12)C(C)C Cc1ccc(F)c(OCC(=O)NCC(C)(C)CNC(C2(CN(C)C)CC2)=O)c1 Cc1c(NC(=O)COc2ccccc2[N+](=O)[O-])cccc1S(N)(=O)=O Cc1ccc(F)c(OCC(=O)N(CC(C)NC(=O)Cc2ccc(Cl)nc2)C)c1 n1(CC)nnc2cc(C(=O)NC(CNC(=O)C=CI)C(C)(C)C)ccc12 N1(C(C(CC)(C)OC)=O)CCC(C2CC2)(NC(c2n[nH]c3c2COC3)=O)C1 O=C1NC(=O)C2(CC(C(=O)N(c3cccc([N+](=O)[O-])c3)c3ccc(F)cc3)C2)N1 c1(C(=O)NC2C(NC(C=CCCC)=O)CCC2)cccc(C)c1C c1(C(N2CCC(O)(C(C)NC(C(CCC)C)=O)CC2)=O)nc2ncccn2n1 c1(C(N(C(CC)CC(=O)NC2CC2c2ccco2)C)=O)cnn2cccc2c1 Cc1cccc(C(=O)NCC2C=CC(NC(C3(CF)CCC3)=O)C2)c1 C(=O)(CCC(C)N(C)C)NC(C)CC1CN(C(=O)CNC2CCOCC2)C1 c1(C(N2CC(N(C(C(CSC)O)=O)C)C2)=O)cc(C)nc(C)n1 Cc1c(Cl)c(C(=O)NC(C2(O)CN(C(=O)C(C#N)C(C)C)C2)C)nn1C C1(CNC(COCCSC)=O)CN(C(c2ccc(=N)[nH]n2)=O)CC(C)(C)O1 C12(C3(NC(=O)C=CBr)CCN(C(CC4CN(C)C4)=O)C3)CC3CC(CC(C3)C1)C2 C1(N(C(=O)Cn2c(C)ccc2C)CC)CCCN(C(=O)CCCN(C)C(C)C)C1 C(=O)(C(C)(O)COC)N1CC(CC(C(=O)NCCC#CCC)F)C1 N1(C(C(c2cn(CC)nc2)(F)F)=O)CC(NC(c2cncnc2)=O)CC2(CC2)C1 C1(NC(COCCN(C)C)=O)CC2CCC1CN2C(C1CCOC(C)(C)C1)=O CN1CCCC(c2cn(CC3C=CCN3C(c3cnc[nH]3)=O)nn2)C1 c1(N2CCC(N(C(=O)CCCCCF)CCC)C2)ncnc2c1nnn2C C1(C(=O)Nc2ccc(Br)c(C)c2F)CCCC12CCN(C(c1cc[nH]c1)=O)C2 c1(C(=O)NCCC(C)N(C(c2c(SCC)nccn2)=O)C)cc(C)cnc1Cl N(C1COc2ccccc21)C(C1N(C(C=CCC)=O)CCC2(CC2)C1)=O c1(OC)c(C(=O)NCCC2(NC(C3CCCN3C=O)=O)CC2)nc(O)nc1O CC(C(=O)NCCc1nc(C(=O)NOCCOCCF)co1)S(C)(=O)=O N1(C(c2c(C)nc(C)[nH]2)=O)CCC2(CCN(C(C3CCN(C)C3)=O)CC2)C(C)C1 c1(CC(N2CCN(C(CC(=C)C)=O)CC2CC(F)F)=O)cccc2ccccc12 c1(C(N2CCN(CC3CN(C(CSCC(N)=O)=O)C3)CC2)=O)cc(N(C)C)ccn1 N1(C(=O)OC(C)(C)C)CCCC(F)(C(=O)N(CCO)Cc2cscc2Br)CC1 c1(C(CNC(C(n2cc(C(C)(C)OC)nn2)C)=O)(C)C)ccc(C)cc1 C1(NC(C(C(C)c2ccccc2)O)=O)CN(C(c2ncc[nH]2)=O)CC2(CCC2)C1 N1(C(CCC#C)=O)CCC(NC(c2cc(O)c3ccccc3n2)=O)C(F)(F)CC1 C1(CN(C(C2CC2C)=O)CC)CCN(C(=O)CCN(C)C(=O)OC(C)(C)C)C1 C1(C(N(CCNC(c2c(C)noc2C)=O)C2CC2)=O)CC2(CCC2O)C1 c1(C(=O)NCC(CCOC)NC(=O)Cc2cccs2)cnn(C(C)C)c1C(C)C C1(COC)CN(C(c2cnc(C)c(N)c2)=O)CCN1C(=O)C=CC1CCCCC1 c1(CC(=O)NC(C(CO)NC(CSCCOC)=O)C)ccc(OCC(C)C)cc1 Cc1oc(C(=O)NC2CC(n3cc(C(C)CCCCO)nn3)C2)cc1Br C(N=c1cc(NCc2ccc(C)s2)nc(C)[nH]1)C1C(CCC)CCCC1 CCCCC(CC)CC(=O)NCC(C1CCCN1C(c1cccc(=O)o1)=O)(C)C c1(C(N(C(C)CNC(C2(C(C)C)CCC2)=O)CC)=O)ccnn1CCC(F)(F)F C(=O)(C1=CC2C=CC1C2)NCc1c(C(=O)NCCC2CC(C)(C)C2)scc1 c1(CN(C(C(=O)N(CC(=C)C)C)=O)C)n[nH]c2c1CCCCC2 C1(C(N2CC(C)N(C(=O)Cn3cnnn3)CC2)=O)COc2ccc(Cl)cc2C1 Cc1ccc(CC(=O)NC2CCN(C(C3CCCC34CC4)=O)C2C)cc1Br Cc1cccc(C(=O)NCC(O)CNC(C2CCC(=O)N2C)=O)c1-n1cccc1 Cc1nc(=N)[nH]cc1C(=O)N(C(C)CNC(=O)CC1CCN(C)C1=O)C N1(c2ncnc3cc(C)[nH]c32)CCC2(CN(C(=O)C(C)N3CCC3)CCO2)C1 c1(C(N2CCC(C(C)(C)NC(C(C)(C)O)=O)C2)=O)ccn2c1CS(=O)(=O)CC2 Cn1cc(-c2oncc2C(=O)NC2CC(C)(CNC(C3(C(F)F)CC3)=O)C2)cn1 c1(C(=O)NCC2C(C)CN(C(c3ncccc3Cl)=O)CC2)ccnc2ccnn12 Cc1cnc(C(=O)NC2CC(C)(CNC(=O)C(C)C(C)(C)C)C2)cc1Br c1(CC)ccnc(C(N2CCCCC2CN(C(=O)Cc2cn[nH]c2)CC)=O)c1 O=C1NC2(C(N3CCN(C(C4CCc5ncnn5C4)=O)CC3)=O)CC3CC1C2C3 C1(CNC(CCc2ccn(C)n2)=O)CC2CCC1N2C(C1CC1C1CC1)=O c1(C(N2C(CNC(c3c(CC)nn[nH]3)=O)CCC2)=O)ccncc1OCC1CC1 c1(C(=O)NCCC2CCC(NC(Cc3cc(COC)on3)=O)C2)nc(O)c(C)s1 C1(C(=O)NC(C=C)C2CC2)CCC(N2CCCCC2=O)CC1 N1(C(c2c(C)cco2)=O)CCC(O)(CNC(C2CCCN2C)=O)C1 C1(C)(NC(c2ccc(CNC(C3CC(C(C)C)C3)=O)nc2)=O)CCCCC1(C)C N1(C(C(C)c2ccon2)=O)CCC2(CC1)CC(C)N(C(c1ccncc1)=O)C2 C(=O)(C(O)CC1CCOCC1)NCCCN(C(C)C)C(c1nncs1)=O c1(CC(C)C)ccc(CC(=O)NCC2CN(C(c3cnccn3)=O)C3CC23)cc1 C1(OC)CN(C(C2(Br)CC2)=O)CC1NC(c1ccnc(CO)c1)=O c1(N(CCCN(C(Cn2c(C)ccn2)=O)C)C)nc2ccc([N+](=O)[O-])cc2s1 C(=O)(C1=CC2CCC(C1)C2)NC(C(=O)NCC1C(C(=O)OC)C1)Cc1cn[nH]c1 Cc1onc(C2CCCC2)c1C(=O)NC1CN(C(C2COC2)=O)C2CC12 N1(C(c2c(OC)csc2)=O)CCCC2CN(C(c3cnc(N)c(Cl)c3)=O)CCC12 c1(OC)cc(Br)c2ccnc(NC(C34CCC(CC3)CO4)C)c2c1 c1(CC)cccc(C)c1C(=O)N(C)CCOCCNC(C1(Br)CC1(C)C)=O c1(CC)c(C(=O)NC(C(N2CCC2(C)C(N)=O)=O)c2ccco2)nnn1C CC1CCCn2cc(C(N3CC(NC(c4ccc(=O)n5c4CCC5)=O)C3)=O)nc21 c1(NC(=O)OC(C)(C)C)ccc(C2C(=O)N2)cn1.C1(CNC)CCN(C(C)=O)C1 C1(CCC)CN(C(=O)CC(C)(F)F)CC1C(=O)NCC1CCC(=O)NC1 C(c1ccc(F)c(C)c1)=CC(=O)NCC1(O)CN(C(CCc2nc(C)sc2)=O)C1 C12(CCC(F)(F)CC1)C(=O)N2.C(=O)(CCNC(=O)CO)NC1(C(C)(F)F)CC1 CC1(C#CC(=O)NCC2CN(C(C3(O)CCOC3)=O)CC23CC3)CC1 CC(C)(C)C(CNC(c1nccs1)=O)C(=O)N1CCC(CC(F)F)C1 N1(C(C)CNC(c2ncc(Cl)s2)=O)CCN(C(=O)Cc2cc[nH]c(=N)c2)CC1 C1(CC#C)CN(C(=O)C(=O)N(c2ccc(C#C)cc2)C)CCC1O.C1CC(=O)N1 C1(CN(C)C(c2cc(Cl)cs2)=O)COCCN1C(c1cccc(=O)o1)=O C1(C(=O)OCC)CN(CC(=O)CC2CCOC2)CC12CC2 c1(C(=O)NCC2C(C)CCN(C(CCOCCC)=O)C2)csc2c1CCCC2 C(=O)(CCC(C)(F)F)N1C(CN(C(c2nc(C)oc2C)=O)C)COCC1 C1(OC)CCC2(C(=O)N(CC(C)C(=O)NC(c3cccnc3)CO)C)CC12 c1(C(=O)NC23C(CN(C(CN4CCC(=O)NC4=O)=O)C2)C3)[nH]nc2ncccc12 c1(CCCC(=O)NCC2CC(NC(C(CC)OCC)=O)C2)ccccc1Cl c1(C(=O)NC(CNC(C2C(OCC)C2)=O)C)c(C)cc(F)cc1C n1(CC(=O)NCC2(OC)CN(C(C3CC3C(F)F)=O)C2)cnc(C#N)n1 N1(C(C(C=C)OC)=O)CC=CC1(C(=O)N(CC(C)SC)C)COC C=CC(CC)CC(=O)NC(CO)CCCNC(=O)CCCN1CCCC1 C12(CC(N3CCC(C)(CNC(CN(CCC)C)=O)CC3)=O)CCCCC1C2(F)F N1(C(CNC(CC(C)C)=O)=O)CC=C(C(=O)NC2CCCCC23CC3)C1 N1(CC)CC(C(=O)NCC(CC(C)C)NC(=O)C(c2ccnn2C)O)CCC1=O C12(NC(c3ccc(OC)c(Cl)n3)=O)CCCC1N(C(c1ccc(N)cc1)=O)CC2 C(C)(CCCCCO)NS(CC(C1CC1)OC)(=O)=O C1(NC(CCC2CCN(C(CN(C3CC3)CC)=O)CC2)=O)CCCC(C)CC1 O(Nc1ncnc2ccsc12)CC(c1ccccc1)CC C1(NC(C2CC(N(C(C3(COC)CC(=O)C3)=O)C)C2)=O)CC(C)CC(C)(C)C1 c1(C=O)ccc([N+](=O)[O-])cc1.C1(CC(=O)N(CC(C)N)C)(COC)CCOCC1 c1(OC)ccc(Cn2nnnc2C2(NCC(N3CC=CC3)=O)CCC(C)C2)cc1 C1(O)(CNC(c2ncc(N(C)C)cn2)=O)CCN(C(C2(CO)COC2)=O)CC1 N1(C(C2(CC=C)CCCN2C(C2CS(=O)C2)=O)=O)CC(C)OCC1C C1(CC(=O)NC(CNC(CCOCC#C)=O)C(C)C)CCc2ccccc2N1 C1(NC(CCC(C)N(C)C)=O)(CNC(c2ccc(=N)[nH]c2)=O)CCCCC1C Cc1cnc(C(=O)NCCN2CCN(C(C3(C)CCC(=O)N3)=O)CC2)cn1 N1(C(C(C(C)C)O)=O)CCC(O)C(NC(c2ccc(F)cc2Br)=O)C1 c1(CC(C)C)cc(C(=O)NC2COCCC2NC(=O)CC2CCOC2)ccc1N c1(C(=O)NC(C(C)NC(CCCC#C)=O)CO)ccc(S(=O)(=O)NCCO)s1 c1(CC)onc(C)c1C(C(=O)NC)N(CCN(C)C)Cc1ccc(Cl)cc1 CC(CNC(C1(c2cccc(C(F)(F)F)c2)CC1)=O)C(F)(F)F CC1(C(=O)NCCC2CCN(C(=O)CC(F)(F)F)C2)CC(F)(F)C1(F)F O=C1NCCN(Cc2c(Br)ccnc2F)C1c1ccc(I)cc1 Cc1cc(NC(C2CC2C(=O)NN2CC3CC3C2C#N)=O)ccc1I.N1CCC1 C1(CN(C(CN(C(C)=O)C)=O)C)CCCC(NC(=O)CSCCN(C)C)C1 S(=O)(=O)(c1ccc(N)c(C#N)c1)NC1CC(C(C)C)C1.N1(CC(C)CO)CCOCC1 CC(CCN(C(=O)C(C)N(C(=O)OC(C)(C)C)C1CC1)CC(F)(F)F)c1cn[nH]c1 c1(C(N(C(C)CCNC(C2CCCS2)=O)C)=O)cnc(O)s1 CC(C)C(Cc1ccccc1)C(=O)N(C1CC2CC1N(C(C1CC(O)C1)=O)C2)C C1(NC(c2ncoc2C2CCC2)=O)CCCN(C(=O)Cc2nc[nH]n2)CC1F c1(C(N(C)CCNC(=O)Cc2cnccc2Cl)=O)cc2n(n1)CCCC2O c1(N(CCCOC)C)ccc(S(=O)(=O)NC(=O)CSCc2nccs2)cc1Cl Cc1c[nH]cc1C(=O)NCc1cc(C(=O)NC(CO)C2(O)CC2)co1 c1(C(=O)NC(CNC(CC(C)SC)=O)C)c(C)ccc(Cl)c1O Cc1nsc(C(N2CCC(CF)(NC(c3ccc(SC4CC4)cc3)=O)C2)=O)c1N c1(OCC(=O)N(CCCNC(c2ccn(C(C)C)n2)=O)CC)c(C)cccc1C C1(c2cccs2)(C(=O)NCCCCCN(C)C(c2nncs2)=O)CCOCC1 CCC(CC)C(C(=O)NC1COCCC1C(N1CCn2nncc2C1)=O)OC C1(CNC(c2cnc(C)s2)=O)CCCCN(C(C2CC(CCF)C2)=O)C1 C(=O)(CCCCCC(C)C)NC1C(CNC(C=Cc2ccc(OC)c(F)c2)=O)C1 Cc1ccccc1C(F)(F)C(=O)N1CC(N(C(=O)C(F)(F)F)C(=O)CC#N)C1 Cn1cnc2ccc(C(N3CCN(C(=O)CC4CCSCC4)C(CO)C3)=O)nc12 CCCC(CCNC(=O)C(C)(C)C1CCCN(C(=O)COC(C)C)C1)CCC c1(C(N2C(CNC(C3(C)COC3)=O)C(C3CC3)CC2)=O)sc2ncccc2c1Cl C(=O)(CC(C)CNC(c1ccc(Cl)cc1)c1nnnn1CCCF)OC c1(NC(c2cc(C)n(C)n2)c2nnnn2C)ccc(Cl)cc1F N1(c2nc(C)cc(C)n2)CC2CCC(C1)C2NC(C1CCCCO1)=O c1(C(CN(C)C)(C)O)cn(C2(C(C3(C(N4CCCC4)=O)CC3)=O)CC2)nn1 c1(CCC)nc(NC(=O)NC2(C)CNC2)cs1 N1(C(CCC=CCC=C)=O)CCC2(CCCN(C(=O)C(C)(O)COC)C2)C1 c1(NCC2C(NC(C=CC)=O)CCC2)c(C)cc(C(=O)OCC)cc1[N+](=O)[O-] c1(C(=O)NC(C)C(=O)NCC(C)CN(C(=O)CC2CCOCC2)C)nocc1Cl CC1CN(C(=O)CCC2CCCC2)CC(C(=O)NOCCN(C)C)O1 c1(C(N(C2CCCC2)CCNC(CCC(C)OC)=O)=O)ccc2occc2c1 C1(C(=O)NC(C#C)CC2CCC2)CCN(C(c2ncn(C)n2)=O)CC1C c1(C(=O)NC(CCOCC)C(=O)NCC(C)(C)CC2CC2)ccc(F)c(C)c1O CC(C)C(CO)N=c1cc[nH]cc1S(=O)(=O)NCCS(=O)(=O)C(C)(C)C N1(CC)CC2CN(C(C3CC(O)CN3C(C3CC(C#N)(OC)C3)=O)=O)CC2C1 C(=O)(CCS(N)(=O)=O)NCCC(C)NC(C(c1c(OC)cccc1)=O)=O N1(C(c2n(C)nc(Br)n2)C(=O)NCCCF)CCC2(COC(C)(C)C2)C1 C1(NC(=O)COC(=O)CCOC(F)F)(CNCc2cccs2)CC2CCC1CC2 C(CCCC(=O)NCC1(C(N2CCOCC2CCOC)=O)CC1)NC(C)=O C1(NC(CC2(C)CC2)=O)CC2CN(C(c3coc(C4CC4)n3)=O)CCN2C1=O Cc1noc(-c2cn(CC(=O)NCCNC(=O)CCCn3cccc3)cn2)n1 CCS(=O)(=O)CC(=O)NC1CC1CNC(C1CN(C(C)C)C1)=O c1(OCC=CCN(C(=O)CC2(C)CCC2)CC)ccccc1C(=O)OCC N1(C(C2(c3ncc(-c4cccnc4F)cn3)CC2)=O)CC(O)CC1C(F)(F)F c1(C(C)C)ncncc1C(N1CC(O)(CN(C)C(c2nnn(C)c2N)=O)C1)=O C1(OC)CCN(C(=O)C(CNC(=O)Cc2cccnc2)N(C)C)CC1C C1(NC(COC(C)(C)C)=O)CCN(C(c2ccnn2C2CC2(F)F)=O)C1 c1(CC)nnc2n1CCCC2C(=O)NC1CC(CNC(=O)CC(F)F)C1 N1(C(C2C(C)(C)CCC2)=O)C2COCC1CC(NC(C1CCC3(CCC3)O1)=O)C2 CC(CC(F)F)C(=O)N(C1(CC(N2CC(O)(C3CC3)C2)=O)CC1)C C1(C(=O)NC2CCC(OC)C2)CC(C)CN(C(c2c[nH]cc2C(C)C)=O)C1 C1(NC(CCC(C)N(C)C)=O)CC2CC(NC(C3CC(O)C3)=O)C1C2 C1(CNC(CC)=O)CN(C(=O)CNc2ccc(C(N)=O)cn2)CCC1(F)F N1(CC(=O)O)CCC(N=c2cc(N(S(N(C)C)(=O)=O)C)nc(Cl)[nH]2)C1 c1(NC(c2nc(NC(CC#C)=O)sc2)=O)c(C)nc2ccccn12 C#CC1CN(C(c2[nH]c(C3CC3)nc2C)=O)CCN1C(=O)C(C1CC1)C1CC1 Cc1cnc(F)cc1C(=O)NC1CCN(C(=O)C(c2ccccc2)O)CC1O C(=O)(C(C(C)C)C(C)C)NCc1occ(C(=O)NC(C(C)SC)C)n1 Cc1ccc(F)cc1C(=O)C(=O)NCC(C1CC1)N(C)C(c1ccnc(Cl)c1)=O c1(OCC)cccc2[nH]c(-c3nc(C)nn3-c3cccc(C(=O)OC)c3C)cc12 C(=O)(C1CCc2cccnc21)NC(C)CNC(c1ccc(F)cn1)=O Cc1cc(C)c(C#N)c(NC2CC(F)(CNC(=O)CCNS(C)(=O)=O)C2)n1 CCCCCCCCC(=O)N1CCCC1CNC(c1cnn(C2CC2(F)F)c1)=O C1(C(=O)NC(c2ncc[nH]2)C)CC12CCN(C(=O)CSC(F)(F)F)C2 N#Cc1ccc(C(N2CCC(CNC(=O)CCN3CCC3)C(O)C2)=O)cc1 N1(C(C(CC=CC)C)=O)CC2(CNC(c3conc3C)=O)CC1CO2 N1(C(c2ccc(N)c(N)n2)=O)CCCC2(CNC(=O)C3=NOCC3)CCCCC12 C12(C(=O)NCC(C3CCCCC3)NC(C(C(C)C)OC)=O)CCC(C)(CC1)CC2 C(=O)(C#CC1(CC)CC1)N(C1CCN(C(C2(C)CCC(=O)NC2)=O)C1)CCC Cc1nnsc1C(=O)NCc1cn(CC(N2CC(OCC(C)C)C2)=O)nn1 N1(C(c2c(C)nc(C)o2)=O)CCC(NC(C2CCCSC2)=O)CC1C c1(N2C(C)C(C(=O)O)CC2)ccc(NC(c2ccccc2)=O)cc1F C1(C(=O)NC(C)CCCCCO)CN(C(c2cnccn2)=O)C2(CCC2)C1 C1(F)(CNC(c2ccn3nncc3c2)=O)CCCN(C(C2CC2[N+](=O)[O-])=O)CC1 N1(C(C(CC=C)(F)F)=O)CCCCC(NC(c2cnn(C)c2COC)=O)CC1 C1(C(N2CCN(C(CC(CC)(C)C)=O)C(CO)C2)=O)CCc2n[nH]cc2C1 CCC(CNC(=NCCc1nccs1)NC1CN(C2CC2)C1)(CC)C(F)(F)F CC1CCC(OCC(=O)NC2CCCCC2N(C)C)CC1 c1(OC)cccc(C(=O)N(C)CC2CCCCN2C(=O)C(C)NC(=O)NCC)c1 CC(O)C(C)C(=O)N(C1CCCC1)CCNC(=O)CNC(=O)CCC1CC1 C(=O)(CCC(=O)NCCCCN(C(=O)C(n1ccc(C)n1)C)C)NCC N1(C(CSCC=C)=O)CCCN(C(=O)CC2CCOCC2)CC1C N1(C(C(C)C2CCCCC2)C(=O)NCC(F)F)CCS(=O)(=O)C2CCCC12 CC(C)C(C)C(C)CC(=O)N(C1CCN(C(c2ccn3c2CSCC3)=O)CC1)C C1(NC(C=Cc2cn(C)nn2)=O)CCN(C(c2cc(C3CC3)nn2C)=O)CC1F Cc1ncccc1CC(=O)NCc1cc(C(=O)NCC(c2ccccc2)O)on1 CC1=NN(C)C(=O)C1CC(=O)N(C(C)CNC(=O)C(O)c1ccsc1)C c1(N2CCC(C)C2)nnc(C(C2CCC2)O)n1CC(=O)NCC(F)F C(=O)(CS(=O)(=O)c1ccccc1C)N(C)CC1(O)CN(C(C(F)=CC)=O)C1 Cc1nc(O)nc(S)c1C(N1CCC(CCN(c2ncc(Cl)c(O)n2)C)CC1)=O Cc1cc(C(N2CCCC(O)(CN(C)C(C3(C)CCCS3)=O)C2)=O)cc(N)c1O C(C(C)(CC(C)C)SC)NC(C(COCC)NC(=O)CSC(C)C)=O C1(C(=O)NCCS(C)(=N)=O)C=CCN(C(c2cn(C3CC3)nn2)=O)C1 N1(C(C(=O)NCCOC)=O)CCC(O)(CN)CC1.C1(C(NC)=O)C(C)(C)C1(F)F C(=O)(C(C)(C)S(C)(=O)=O)N1C(C2(NC(C3CCC(CC)O3)=O)CC2)CCC1 Cc1cccc(C2(C(N3CCC(F)(CNC(c4cc(C)sn4)=O)C3)=O)CC2)c1 N1(C(=O)Nc2ccc(CN(C)C)cc2)CC2C=CCOC2C1 C(CCCCCNC(C1(CO)CCCO1)=O)NC(=O)CN1CCOC1=O C(c1cccc(Cl)c1)=CC(=O)NCC1C2CN(C(c3ccn(CC)c3C)=O)CC21 Cc1ccc(F)cc1CC(N1CCC(C2CCCN2C(C23CC(C)(C2)C3)=O)C1)=O c1(C(N2CCCC(NC(C(CC)(CC)OC)=O)C2C)=O)cn(C)c(=O)nc1O C1(C#N)(C(N2CCC(C(N(C(C)C3CC3)C3CC3)=O)C2)=O)CC(=O)C1 C#CC1CN(C(=O)Cc2cncs2)CCN1C(=O)C1=COCCC1 N1(C(C(C)(C)OC)=O)C2COCC1CC(NC(C1CC1c1cccnc1)=O)C2 C(=O)(CC(C)CCC=C(C)C)NCC(CC(C)C)NC(Cc1ccc(SC)o1)=O N1(CCN(Cc2cccc(C)c2)Cc2cccs2)CCC2COCCC12 Cc1scc(C(=O)NC2(CO)CCN(C(=O)C(c3ccc(Cl)cc3)O)C2)c1N C1(NC(c2cc(C)ncc2)=O)CN(C(c2cc(=O)c(Br)c[nH]2)=O)CC2(CC2)C1 c1(C(N2CC(OC)C(NC(C3C=CCC3)=O)C2)=O)cccc2[nH]c(=N)oc12 c1(OC)cc(C(N2CCC(N(C)C(C3CCCCS3)=O)CC2)=O)cc(F)n1 C1(C(N2CCC3(CCCO3)C2)=O)Cc2cc(O)ccc2CN1Cc1nccs1 O=S(=O)(C=Cc1ccccc1)NCC1(F)CCCN(Cc2ccncc2F)C1 c1(C(=O)NCC(CC)N(C(=O)CCOCC(C)(C)C)C)c[nH]nc1COC N1(C(C2(C)CN(C(C3CC3(C)C)=O)C2)=O)CCC2(CNC(=O)N2)C1 C1(C(=O)NC2CCN(C(C)C)C2=O)CCC(C)N(C(C2C(C(C)=O)C2(C)C)=O)C1 CC1CN(C(c2cnn(CCF)c2)=O)CC(CCNC(C2(O)CCC2)=O)O1 C1(C(N2CC(OCC(C)C)C2)=O)CC(C)CCN1C(=O)C(C)C(=O)OC.CO C1(NC(COC2C(C)CCCC2)=O)CCN(C(=O)CCC(F)F)CC1F C12(C(=O)NCCC3N(C(C4CC(F)(F)C4)=O)CCCC3)CCC(O)(CC1)CC2 Cc1ccc(O)c(C(N2CCCC(NC(=O)C(F)n3ccnc3)C2)=O)n1 C=CCCC(C)(C)C(=O)NCC12CC1CN(C(c1ncc[nH]c1=O)=O)C2 c1(C(C)C)onc(C2CCCO2)c1C(=O)NC12CC(C)C1C2.C12CCC1NC2=O c1(C(=O)NC2CCC(CNC(C3C(CC)OCC3)=O)CC2)ccc(C#N)cc1F c1(C(=O)NCC(C)N(C(=O)CN(CC)CC2CC2)CCC)ccccc1C c1(OCC(=O)NCC(CNC(c2ncc(C(F)F)s2)=O)CO)cccnc1Cl CN1CCC(NC(=O)CC(CC2CC2)NC(c2csnn2)=O)C(C#N)C1 N1(C(C(=O)NCCC(=C)CNC(=O)CS(=O)(=O)NC)C)CCc2ccccc2C1 C1(C(C(=O)NCCOC(CC)(C)C)C)CCN(C(c2nnn(C)c2N)=O)CC1 C1(F)(C(=O)NC(CCCC)CNC(=O)CSC(F)(F)F)CC2(CCC2)C1 C1(CNC(c2cccc(N(C)C)n2)=O)CN(Cc2cccnc2)CCC1(F)F Cc1cnn(C(C)C)c1C(=O)NCC1CCCN(C(C2CCC23CCC3)=O)C1 C#CCC(C(=O)NC(CCSC)C(=O)Nc1ccc(CO)nc1)C1CC1 Cc1cc(C(=O)NCC2CCC(NC(C3(C)CCNC(=O)C3)=O)C2)cnc1O C1(C(N(C)CC2CCCC2NC(=O)Cc2ccno2)=O)CCNC(=O)C1 C1(NC(C(CSC)O)=O)COC2(CCN(C(C3(F)CCC(F)(F)CC3)=O)CC2)C1 C1(C(=O)Nc2c(OC)nc(Cl)cc2)CN(Cc2ccnc(Cl)c2F)CCC1(F)F c1(C(=O)NC(C)CN(C(=O)CN2CCCC2)C)cnc(N)c(-c2ccccc2)c1 C(=O)(C(O)C(F)(F)F)NCc1cn(CC(C)NC(Cc2cnc(C)s2)=O)nn1 C1(CC(=O)NC2CCC(CN=c3[nH]nc(C(C)(C)C)o3)C2)Cc2ccccc2O1 N1(C(C(C)SCC)=O)CC2(CC(NC(c3csc4cncn34)=O)CO2)C1 N1(C(C2(C(C)C)COC2)=O)CC2ON=C(CNC(=O)CSc3cccnc3)C2C1 CC(C)C(C(=O)NCC1CC(C)CN(C(=O)CCOCCN(C)C)C1)C(C)C c1(C(=O)NC(CN(C(=O)CCOC(C)C)CC)C)cc(Cl)c(Cl)cc1N N1(C(C2N(C(c3cc(C)n(C)c3)=O)CCN(C)C2)=O)CC2(CCC(=O)NC2)C1 N1(C(Cn2c(C)cc(C)n2)=O)CCC(F)CC1C(=O)N(CC(Cl)Cl)C C(=O)(C#CC1CCCC1)NC12C(CN(C(c3cccc(C#N)c3)=O)C1)C2 CCCC(C)C(=O)NCCN(C(C1CC(C(=O)OC)(OC)C1)=O)CC1CC1 C(=O)(C(CC(C)C)ONC(=O)CC(C)O)N1CC(OC)C(OC)C1 C1(C(=O)NC2(CNC(c3cc4[nH]ccc4s3)=O)CC2)CCn2nnnc2C1 C(=O)(C1=Cc2cc(F)ccc2OC1)NCC1C2CN(C(C=C(CCC)C)=O)C1C2 c1(C(=O)NCC2C3CN(C(C(CC)NC(N)=O)=O)C2C3)ccccc1[N+](=O)[O-] Cc1ccc(C(=O)NC(C)C(CO)NC(c2ccc(C#N)o2)=O)cc1C(C)(C)C N1(CC(N2CCC(C)C2CNC(c2ccc(F)o2)=O)=O)CCC(=O)NC1=O C1(NC(c2ccc(COC)cc2)=O)C2CCC1CC(NC(C1CCCCS1)=O)C2 c1(C(C(=O)NC)N(CCC(N)=O)C)ccc(OCc2ccccc2Cl)cc1 CCCC(C)C(=O)N1CCC(O)C1C(=O)NC(C)CN(C)C C(=O)(C(=O)C(C)CC)NC(C(=O)NC(CC)C(N)=O)CCF CCCCCC(O)C(=O)NCC1CCC(CNC(c2cc(N)cc(F)c2)=O)CC1 C12(C(=O)NC(N=S(C)(C)=O)=O)CC(CO1)N(Cc1ccc(N3CCCC3)cc1)C2 C(CN=c1[nH]cnc2cccc(Br)c12)(C1CC1)NC(c1ncc(C)c(Cl)c1)=O C(=O)(C1=CCCCO1)NC(CC=C)C(=O)N(c1ccc(C)cc1)CC(=O)OCC CC1(C)CCC2(CN(C(c3ccc(-c4nnc(S)o4)cc3)=O)CCO2)C1 Cc1c(C(=O)NCC2C=CCN2C(=O)CCCn2cccn2)ccc2cncn12 N1(C(C(CC)OC2CCCC2)=O)CC(NC(c2cc(CC(C)C)[nH]n2)=O)C(C)C1 N1(C(C2(NC(=O)OC(C)(C)C)CCC2)C)CCCN(c2ncc(F)cn2)CC1 Cc1cnc(CC(=O)NCc2csc(CNC(=O)Cc3ccoc3)n2)[nH]1 C(c1ccc(OC(=O)C(C)CS(C)=O)cc1)=CC(=O)OC c1(NC(C2(NC(C3CC=CC3)=O)CC2)=O)cccc(C(F)(F)F)c1 c1(C(=O)NCCC2CCN(C(C(CC)(C)C)=O)C2)ccc(C#N)c(C)n1 c1(C(N(CC(CNC(c2scc(C)c2C)=O)O)C)=O)cc2ccccn2n1 C1(NC(CC2CCCC(=O)C2)=O)CN(C(c2cc(=O)cc[nH]2)=O)C2(CCOC2)C1 C1(C(=O)NC(CCOC)(C)C)CCN(C(=O)C(C)(C)CSC)C(C)(C)C1 c1(NC(c2cn(-c3cccc(OC)c3)nn2)=O)c(Cl)ncc(Br)c1C N#Cc1ccc2c(c1)CCC2NC(=O)Nc1ccccc1-c1cccnc1 C1(C(N(CC(=O)NC)CC(=O)OC)=O)CCOC1c1nccn1CC(C)(C)C C1(C(C)NC(=O)CC2(C)CCN2C(C)=O)CCN(C(=O)CC#N)CC1 C1(C(N2CCCC(NC(c3c(CC)nc(=N)[nH]c3)=O)C2)=O)CCC2(C1)CC2(F)F CC1CN(C(C2CCCO2)=O)CC1NC(=O)C=CCOc1ccccc1 N1(C(CC(CC)NC(=O)Cc2cccnc2)=O)CCC12CCOCC2 S(=O)(=O)(c1ccc2nn[nH]c2c1)NC(C1C(c2cccc(C)c2)C1)=O N1(C(C(CCC)OC)=O)CC2CCCC(N(C(=O)COC3CCOC3)C)C2C1 N1(C(c2cccc(F)c2F)=O)C2CCC1CN(CCc1cc(Cl)ccc1Cl)CC2 C12(C(=O)NCC3=NOC(C)C3)CCCC1CCN2C(=O)COc1ccsn1 c1(C(=O)NCC(C)(C(C)C)NC(C=CSC)=O)ccnc2c1cnn2C CCN=c1[nH]c(C)c(C(=O)NC2CC(C)N(C(=O)COc3cnn(C)c3)C2)s1 c1(C(=O)NCC2CCN(C(c3nc(C(C)(C)C)sc3)=O)C2)ccc(NC=O)cc1 c1(NC(C2C3CN(C(c4c(CCC)[nH]cc4)=O)CC32)=O)ccc(F)cc1C c1(C(=O)NCC2C3CN(C(c4c(C)nn(C)c4)=O)CC32)c(C)nn(C)c1Br C(=O)(C1CCCc2nnn(C)c21)NC(C)CNC(c1ccc2oc(O)nc2c1)=O c1(COC)nc(OC)cc(NC(C)CC(C)NC(=O)CN2CC(=O)NC2=O)n1 N1(C(=O)C=Cc2ccoc2)CC2CC2(C(=O)Nc2csnc2C2CC2)C1 CCC(CC)(CC)C(=O)NC1CCCCC1CC(=O)NC(C)Cc1ccco1 Cc1cncc(C(N2CC(CC(=O)NCCn3ccnc3C)CC2C)=O)n1 C1(C2CCN(C(=O)CCCn3ccnc3C)C2)(NC(C=CCCC)=O)CC1 C1(CCC(=O)NC2CC(CNC(CCN(C)CC)=O)C2)CCC(C2OCCO2)O1 C(C)(C(=O)NN1CCCC1C(N1CCN(CC(C)O)CC1)=O)SCC C1(CNC(c2cocc2Br)=O)COCCN(C(=O)Cc2cncnc2)C1 CC1OCCN(C(=O)CCS(C)(=O)=O)C1C(=O)Nc1ccc(O)c(CO)c1 CCC(CC)C(C)C(=O)NCC(c1ccc(F)cc1)NC(c1snc(Cl)c1Cl)=O C(=O)(N=c1ccn(C2CC2)[nH]1)C1C(NC(c2c(C)cccn2)=O)CCCCC1 C(=O)(NNC(=O)N(CCOC)CC1(OC)CCSC1)SCCC N1(C(Cc2cc(C)no2)=O)CC2C=CC1C(C(N1CCCC(C)(F)C1)=O)C2 C1(C(=O)NC2CN(C(C3CCCCC3)=O)C3CC23)CC2(CCC2)CO1 C1(CNC(Cc2cc(C)ns2)=O)CN(C(c2cc(C(N)=O)n(C)n2)=O)CCC1C N1(Cc2c(OC)nc(Cl)cc2)C2CCC1CN(c1ncc(Br)c(OC)n1)C2 Cc1oc(CNC(=O)COc2cccnc2)nc1C(=O)N(CCCO)CCCF C(c1cnccc1C)=CC(=O)NC1C(CNC(CC(COC)C)=O)C1 c1(SC)cc(C)ccc1C(N1CC(C)(NC(c2csc(-c3cnc[nH]3)n2)=O)C1)=O Cc1ncnc(O)c1C(N1CC(NC(C2(C(F)F)CC(F)(F)C2)=O)CC(O)C1)=O c1(C(C(=O)NCC(CNC(=O)CC2COCCO2)O)(F)F)ccc(F)cc1 Cc1noc(C)c1C(C)CC(=O)NCCCOCCNC(=O)Cc1cccn1C Cc1ccc2c(CNC(C3CCCCCN3C(=O)OC(C)(C)C)=O)ccnc2c1 c1(-n2cc(CNCC3C(CF)C3)nn2)ccc(Cl)c(N)c1 CCN(OC)C(=O)CN=c1[nH]c(=NC(C)C2CCOC2)[nH]c2ccsc12 c1(C(N(C2CCCC(NC(c3nn(C)cc3Cl)=O)C2)C)=O)cn2c(n1)COCC2 c1(C(N(CCNC(=O)CC23CCCC2C3)CC)=O)ccc(Cl)c(-n2nnnc2C)c1 c1(C(=O)OCC2CC2)ccc(CN2C(=O)CC(C(C3CC(F)(F)C3)O)C2)nc1 c1(C(=O)NC(CC)CN(C)C(C2CC(OC)C2)=O)c(C)sc(C)c1C#N C1(CN(CC)CC)CCN(C(=O)NCc2cccc(-c3cccs3)n2)CC1 C1(C(=O)NC(c2ccc(F)cc2)COC)CCCN(C)C1=O N1(C(C2(c3cc(C)no3)CC2)=O)CC2CCCC(NC(=O)C(C)(C)CF)C2C1 C1(CNC(=O)CCF)CN(C(=O)CCN2CCCCCC2)C2CCN1C2 C1(C(=O)NC(CCOC)(C)C(=O)O)CC(=O)OC12CCCCC2 S(=O)(=O)(C1CC1)NCC1CN(C(=O)COC(CO)CCc2ccccc2)C1 c1(C(=O)NCCCN(C(C2CCCC(C)C2)=O)C)csc2ncnc(O)c12 CN1CCN(CCC(N2CCC(CNC(=O)C3=CCSC3)CC2)=O)CC1 c1(OCC=C)cc(Cl)ccc1C(=O)NCCC1CN(C(c2c(O)noc2C)=O)C1 c1(NC(CC2CCC(NC(Cc3c(C)n(C)cn3)=O)C2)=O)cccc(Cl)c1C N1(C(c2cc(OC)ncc2)=O)CC2CCN(C(C3(CCF)CC3)=O)CC2C1 c1(CC)cc(C(=O)NC(CC2CC2)C(=O)NCc2nc(C3CC3)n[nH]2)ccn1 C12(C(=O)NC(C3CCCC3)C#C)CCCC1CN(C(C1CCC(C3CC3)C1)=O)C2 N1(C(C2COCCOC2)=O)CCC(C2(O)CN(C(C3(O)CCOC3)=O)C2)CC1 N1(C(CCC=C)=O)CC(C2CCN(C(c3ccc(OCC)cc3)=O)C2)C1 C(C(C)CN(C)C(C1CC(N(C)CC)C1)=O)NC(C1(CC=C)CC1)=O N1(C(C(=O)NCC(C#C)OC)=O)CC(C(F)F)(OCC)C1 N1(C(Cc2cc(OC)c(O)cc2)=O)CC2(CC1CNC(C)=O)CC2(F)F C1(NC(C=CC(=O)OCC)=O)CCOCC1NC(C1CC2CC2C1)=O c1(C(N(CCNC(C2CCC(C(C)C)CC2)=O)C)=O)cc(F)c(F)cc1O c1(NC(c2ccc(-c3ccc(Cl)cc3)o2)=O)ccc(-c2cccc(F)n2)cc1F c1(CC)ccccc1CC(=O)N(CC(O)CNC(c1sc(N(C)C)nc1Cl)=O)C c1(C(=O)NC23C(CN(C(c4c(C)nc[nH]4)=O)C2)CC3)cc2n(n1)CCCC2 C1(NC(C=C(CC)C)=O)C2CCN(C(C3(c4c(Cl)cccc4Cl)CC3)=O)CCC12 c1(-c2cn(CCC(=O)NCC(C)(C3CC3)OC)nn2)ccc(CC2CCC2)cc1 N1(C(C2(N(C)C)CCOCC2)=O)CCCCC(NC(C2(C)CCCNC2=O)=O)C1 NS(=O)(=O)c1ccc(C(=O)Nc2ccc(-n3c(=O)oc4ccccc34)cc2)o1 N1(C(C(C)=C2CCC2)=O)CCCC1(C)CNC(c1ocnc1C(F)(F)F)=O Cc1noc(C)c1C=CC(N1CC(NC(C2CCCC(F)C2)=O)C1)=O N1(C(C(CNC(c2cnnn2C)=O)OC)=O)CCCC(O)(CO)C1 Cc1c(C(=O)NCC2(C(=O)NC3CC4C(C3)C4(F)F)CC2)c[nH]c1C#N C1(c2nc(C(C)C)[nH]n2)CCCCN1C(c1ccnc(OCC2CC2)c1)=O S(=O)(=O)(c1cc(C(N2CCCCC(CNC(C3(C)CCC3)=O)C2)=O)c(C)o1)NC C1(NC(Cn2ncc(C)c2)=O)C2COCC1CC(NC(=O)C(C)n1cccn1)C2 c1(CN(C(c2cn(C)nc2Br)C(=O)NC(CC)C)C)cc(Cl)ccc1F c1(C(N2CCCC2CCOC)C(=O)NC(CC)C)ccc([N+](=O)[O-])s1 C1(C)(NC(C2(CNC(C(C)OCCOC)=O)CCCO2)=O)CCCC1(C)C C12(C(=O)NC(C)(C)CCNC(=O)C(C3CC(F)(F)C3)O)CC1CNC2=O N1(C(c2cccc(C)n2)=O)CCC2CCCC12CNC(c1cccc(C)c1F)=O c1(C(=O)NC(C2CCN(C(c3nc(OC)c(C)s3)=O)C2)C)c(C)ccnc1O c1(C(C(=O)N(CCCN(C)C(C2C3CC4C(C3)C24)=O)C)C2CC2)ccc(F)cc1 N1(C(c2ncsc2C)C(=O)OCC)CCCC(n2nccn2)C1.C(CCO)S N1(C(C2(OC)CCOC2)=O)CCC2(C1)CN(C(c1ccn(C3CCCC3)n1)=O)C2 c1(CC2(C(=O)SCC(=O)NCCN(CCC)C(C3CCC3)=O)CCC2)cc(C)no1 Cc1conc1CC(=O)NC1CC(O)C1CC(=O)N(c1cnn(C)c1)C(C)C CC(O)C(F)(F)C(=O)N1CC(N(C)C(c2sccc2SC(=O)OC)=O)C1 C12(NC(c3cc(C(C)C)[nH]n3)=O)CCOCC1CN(C(=O)C=Cc1cscn1)C2 Cc1cc2c(C(=O)NC3CC3CNC(c3c(Cl)n[nH]c3C)=O)cccc2o1 C(=O)(C(CC(F)F)NC(c1cc(Cl)n(C)n1)=O)N1C(C(C)C)CC1 C1(CC)CCN(C(=O)NN(CCC2CC23CC3)Cc2ncoc2C2CCC2)C1 N1(C(CSCCOC)=O)CCC2(CCN(C(C3CC(O)CN3C)=O)C2)C1 C(C)(CC(=O)NCCC1(CNC(c2cc(C(F)F)no2)=O)CC1)=C(C)C C1(NC(c2cc(CNC(c3c(CC)onc3C)=O)ncc2)=O)CCCCCC1F CC(C)C(F)(CNC(=O)CCCC1CCCO1)C(=O)NOCCO n1(CC)nc(C)c(C(=O)NCC(CC(F)(F)F)NC(C2CCCCO2)=O)c1Cl CC1(NC(=O)NCC(O)COc2ccccc2Cl)CCCOC1 N1(C(c2cncc(OC)n2)=O)CCn2ncc(CNC(=O)C=C(C)C)c2C1 c1(CN2CC(C)(OC)C2)ccccc1Cl.C1(=O)C(c2ccsc2)N1 C(=O)(C(CC(C)(C)C)OC(C)=O)NCC1C(CC)CCN1C(=O)C(C)N1CC(C)C1 N1(C(c2ccc(C)c(O)c2)=O)C2CC(F)C(C2)C1C(=O)NC1CC(F)C1 N1(C(C(C)CC=Cc2ccccc2)=O)CCCN(C(c2cc(Cl)cs2)=O)CC1 C1(C(=O)N(C)Cc2ccns2)(COC)C=CCN1C(=O)Cc1nocc1C N1(C(C(=O)NCC)=O)CC(NC(C23CCCC2(C(N)=O)C3)=O)CC12CCOCC2 C(c1ccccc1Cl)=C(C)C(N1CCN(C(C2C(C)C2C)=O)C(C)C1)=O CC1=NS(=O)(=O)NC(C)=C1CCC(=O)NCCCNC(C1(c2ncco2)CC1)=O CC(C)CS(=O)(=O)CC(=O)NCC1CC(CNC(C2C=CCC2)=O)C1 N1(C(=O)Nc2ccc(CC)cc2)CC2CCC(C1)C2NC(=O)C1CC1 CC1CC(C(=O)NCC(c2cnn(C)c2)C)CCN1C(C1CCCCC1)=O CCC(C(=O)N1CC(SCC(=O)NC(c2cccs2)C)C1)SC.C(C)(C)S Cc1cnc(CN2CCNCC2C(=O)Nc2ccccc2)c(Br)c1 C(CC(CNC(C1(C(C)(F)F)CCC1)=O)NC(=O)C=CC(F)(F)F)OC C12(CNC(c3ccccn3)=O)CCCCC1N(C(c1n[nH]c3c1CCC3)=O)CC2 CC(F)(C(=O)NC1CCCN(c2nccnc2Cl)C1)C(F)(F)F CN1CCN(C(c2cccc(C3CC3)c2)=O)C(CNC(=O)Cc2cncn2C)C1 N1(C(c2cnc(C)[nH]2)=O)CCC2(NC(C3CN4CCCN3CC4)=O)CCCCC12 S(=O)(=O)(c1cccc(Cl)n1)N1CC2N(C(c3cc(C#N)c(F)cc3)C3CC3)C2C1 N1(C(Cc2cc(C)[nH]n2)=O)CC2CC1CN2C(=O)CC(C)c1ccco1 c1(OC)ccccc1OCCN(C(=O)C(=O)NCC1NCNC1(C)C)C c1(OC(C)C(=O)NC(C2(O)CN(C(=O)C(CO)c3cnc[nH]3)C2)C)ccccc1 C1(NC(c2c(C)cccc2C)=O)CCC2(CC1)CC2NC(c1ccc(C#N)s1)=O c1(C(N2C3CC(NC(COC(CC)C)=O)C(C3)C2)=O)cnc2ccccc2n1 Cc1cc(C(=O)N(CCCC(=O)NCC2CC2(Cl)Cl)C)c(N)s1 c1(C(=O)NC2CC(CNC(C(C)C3(O)CCC3)=O)C2)cc2cn[nH]c2cn1 N(C(=NCCN1CCCOCC1)Nc1ccc(C(=O)OC)cc1)CCC(=O)NC N#CCC(CC(=O)N1CCOC(c2cccc(F)c2)C1)c1ccccc1 N1(C(C(C)O)=O)CC2CCC2(CNC(=O)C=Cc2cccc(OCC#N)c2)C1 c1(C(=O)NCC=CCNC(=O)COC2CCOCC2)ccc2c(O)nccc2n1 N1(C(C(C)N2CCC2)=O)CC(O)(C(F)C(=O)NC2CC=CC2)C1 C1(C(=O)NCCCN(C(Cn2cc(C(=O)OC)nn2)=O)C(C)C)CC(C)C1(C)C Cc1cccc2c(C(N3CC4CCN(C(=O)C(O)C(C)C)C4C3C)=O)csc12 N1(C(C=CCCC)=O)CCN(C2CCC(NC(c3cc[nH]c3CC)=O)C2)CC1 N1(C(CC2(CSC)CC2)=O)CCCC2(CCN(C(=O)C(C(C)O)N(C)C)C2)C1 C1(C(=O)NC(CSCC)C(=O)N(C2CCC3(CC2)CC3)C)CC(=O)NC(C)C1 C1(C(=O)NCC(C)(O)C2CCC2)CSCN1C(C1CCCCO1)=O N1(C(Cc2ccc(C)nc2Cl)=O)CC2CCC1CN2C(=O)CCSCC(C)C n1(CC)nc(C)c(C(=O)NC(C2(O)CCN(C(c3cc(Cl)c(Cl)s3)=O)C2)C)c1Cl N1(C(CCCSC)=O)CCC(F)C(NC(c2ccc(C(=O)OC(C)(C)C)cc2)=O)C1 c1(CCCC(=O)Oc2cc(Cl)ncc2F)ccc2c(c1)OCCO2 C1(CNC(c2cc(C)c(C)s2)=O)CN(C(c2cncc(N)n2)=O)CCC1C c1(C(=O)NC(CC)CNC(c2cc(O)n(C)n2)=O)nccn2c(Br)cnc12 c1(-n2c(C)nnn2)cccc(C(=O)NCC(C2CCC2)NC(=O)COCCF)c1 CC1CC(=O)NC1C(=O)N(CCCCN(C)C(C1(C(F)F)CCOCC1)=O)C Cc1c(O)ccc(C(N2CC3(C2)CN(C(=O)CN(S(C)(=O)=O)C)C3)=O)c1C C1(NC(C2C(C)(C)CC2)=O)CCCCCN(C(=O)COCc2ccccn2)C1 C(C1CN(C(C2CCSC2)=O)Cc2ccccc21)NC(c1nn(CC)c(C)c1)=O Cc1ccc2c(c1)CCC(C(N1CCN(C(=O)C=Cc3cc[nH]n3)C(C)C1)=O)O2 CCC(C)C(C(=O)NCC(O)CC(F)(F)F)NC(=O)CCNC(=O)CO CCC(F)(F)C(=O)NC1CCCC(CN(C(=O)C=Cc2cc[nH]n2)C)C1 N1(C(CCS(C)=O)=O)C2COCC1CC(NC(C1CCCN1C(N)=O)=O)C2 S(=O)(=O)(c1ccc(C)c(C)c1)N1CCC(CNC(c2c(OC)ccc(Cl)c2)=O)C1 c1(C(=O)NCC2(CNC(CCC(C)SC)=O)CC23CCC3)ccnc2cc[nH]c12 Cc1ccccc1C=CC(N1C(C(=O)NCCNC(=O)N(C)C)CCC1C1CC1)=O C(=O)(C(CNC(C1(C)CCC(=O)C1)=O)C(C)(C)C)NCc1c(C)cc(C)s1 Cn1cc(NC(C2CCN2C(=O)C(c2ccc(F)cc2)=O)=O)c(C(F)(F)F)n1 CCCC(C(O)C(=O)NC1CC(C2CCC2)C1)NC(C1CS(=O)(=O)C1)=O N1(CC)CCOCC1C(=O)NC1CC(F)(CNC(=O)CC2CCOCC2OC)C1 C1(S(C)(=O)=O)(C(=O)NC2CCCC(N(C)C(c3n[nH]cc3Cl)=O)C2)CC(O)C1 c1(C(=O)Nc2cc(C)c(NC(C3CC34CC4(F)F)=O)cc2)cccc2ncsc12 N1(C(C23CCC(OC)C2C3)=O)CCC2CCCC12C(N1CCC(F)(F)CC1)=O C(=O)(CC(C)(C)CCC)N(CC(=O)NC1(C(=O)OCC)CC2CCCC12)CC#C c1(C(=O)NC(CC)CNC(=O)CC2(OC)CC2)cccc(-c2nnco2)c1 C=CCC(CNC(=O)C(CC)CC=CC)C(=O)NC1CCC=CCC1 C(=O)(CCC(C)(C)[N+](=O)[O-])NCC1CC(C)N(C(=O)Cc2nncn2C)C1 C1(CC(=O)NC(C)CN(C)C(C)C)(OCC)CN(C(=O)C(C)COC)C1 CC1CCCN(C(c2cccc(CO)c2)=O)C1CCNC(C1(O)CC(CF)C1)=O Cc1nn2cc(C(N3CC(C)N(C(=O)C(C)OCCN(C)C)CC3C)=O)nc2s1 N1(C(C2C(=C)CC2)=O)CC(C(F)(F)F)CC1CNC(=O)CCc1nc(CC)no1 N1(C(C=CCC(C)(C)NC(c2c(CC)con2)=O)=O)CCC2CCN(C)C2C1 C1(C(=O)NCC(C)(C)CNC(C2(O)CCSCC2)=O)CCC2(CCCCC2)C1 C1(NC(C(C(CC)C)OC)=O)C(C)CCN(C(C2CN(C)C(=O)N2)=O)C1C c1(C(=O)NCC(CNC(Cc2c(C)cco2)=O)(C)O)csc2c1CCCC2 c1(C(CN(C(Cn2cc(C3(N(C)C)CCC3)nn2)=O)CCO)O)cccc(Cl)c1 c1(C(=O)NC2CC(CNC(c3nc(CC)oc3)=O)C2)ccc(OCOC)cc1 Cc1cc(OCCCN(C(C2CCc3cnn(C)c3C2)=O)CC)ccc1[N+](=O)[O-] Brc1ccc2c(c1)CCC2c1noc(-c2cn(C3CCOC3)nn2)n1 c1(C(N(CC(CC)NC(=O)CCCF)CC)=O)n[nH]c(C2CC2)c1C C=CC(C)(CC)NC(c1cn(CCNC(C2CCO2)=O)nn1)=O c1(C(N2CCC(N(C(C3C=C(C)CS3)=O)CC)C2)=O)sc(C)cc1C N1(C(C=C(C)C(C)(C)C)=O)CC2CC2C1CNC(=O)COC1CCN(C)CC1 CCC(C)(CNC(c1ccon1)=O)C(=O)N(C1CCN(C(C)C)C1)C c1(C(C)=O)cc([N+](=O)[O-])ccc1NC1CCC2CN(C(=O)C3=C(Cl)CC3)CC2C1 Cc1cc(C(N2CCN(C(=O)C(C)O)C(CC(F)F)C2)=O)ccc1C1CC1 N1(C(c2ncn(C)n2)=O)CC(CNC(=O)C=Cc2ccncn2)C(C(F)(F)F)C1 CONC(=O)C(=O)N1CC(O)CC1C(=O)N(C(C)C(C)C)C CC(=O)C(C)CC(C)C(=O)NCc1n[nH]cc1C(=O)NCc1snnc1C C1(O)(CNC(CCN(CC=C)C(C2CCS2(=O)=O)=O)=O)CCC(C)CC1 c1(CCC)ccc(C(=O)NC2C=CCN(C(c3cn(CCC)nc3C)=O)C2)cc1 C1(NC(c2c(CCC)nns2)=O)CN(C(c2ccccc2Cl)=O)CCC1C C(CC(O)CCO)NC(C1CN(C(=O)C(F)C2CCCC2)CCO1)=O C1(S(C)(=O)=O)(C(=O)NC(C(C)C)CNC(=O)C(C)(C)N(C)C)CCCCC1 c1(N(C)Cc2cc(-c3c(OC)cc(F)cc3)ncc2)c[nH]c2c(Cl)cccc12 C1(CNC(C(C(C)C)NC=O)=O)N(C(=O)C(O)C2CCC2)CCCC1(C)C C1(C(=O)NC(C)(C)CO)CC2C=CC1N(C(=O)Cn1cnnc1O)C2 c1(OCC)ccc(C(N2CCC(NC(C3CC3C)=O)C(F)C2)=O)cc1Cl CC1CCC(CNC(=O)Cc2ccco2)CN1C(C1CCC(C)(C)O1)=O c1(C(=O)NC(CCNC(C(C)OCC#C)=O)C)conc1-c1ccccc1 c1(C(C(=O)NCC2(CNC(C34CCC3CC4)=O)CC2)O)cccc(Br)c1 C1(C)(C(=O)NC(CC)CNC(c2coc(COC)n2)=O)C=CCCC1 c1(NC(C2(SC)CN(C(c3cc(OC)cs3)=O)C2)=O)ccc(F)nc1 CC1OC(=O)NC1C(=O)N(C)CC1CCCC1NC(=O)CCC1CC1(C)C C1(N(C(C(c2ccccc2F)C)=O)C)CN(C(=O)CCP(C)(C)=O)CCC1C N1(C(c2c(C)con2)=O)CCN(CCNC(=O)CC2CCC(=O)O2)CC1 CC1(CCCOC2CCC2)CCCN1C(C1(c2ccc(Br)cc2)CCCCO1)=O CC1(C)CCC(C(N2CCC3CCC23CNC(c2csnn2)=O)=O)CC1 C1(NC(CCCn2c(C)ncc2)=O)CN(C(C2CC3CC2C3)=O)CCC1C C1(C(=O)NC2(CO)CN(C(C34CC(C)C3C4)=O)C2)CC2(C1)CC(O)(C(F)(F)F)C2 C1(C)(C(=O)NCC(CC(=O)NCCCC2CC(C)C2)OC)CCC(O)CC1 C(CC(C)(C)CC(=O)N1CCN(C(=O)C2=CCCOCC2)CC1CCO)OC c1(C(N2C(CC)C(C(=O)NCC3C(C)C3C)CC2)=O)ncc(N)cc1C C#Cc1ccc(Cl)c(C(N2CC(NC(C3CCn4cncc4C3)=O)C(O)C2)=O)c1 c1(NCC(=O)NC2(c3ccc(Cl)s3)CC2)cc(F)c(F)cc1Br c1(CN(C(c2sccc2I)C(=O)NCc2cccs2)C)cccc2ccccc12 c1(C2C(C(=O)NC3CC(CCNC(C)=O)C3)C2)ccn(C)c1 N1(C(CN(C2CCCC2)C)=O)CCC2OCCN(C(c3ccc(=O)oc3)=O)C2C1 Cc1ccc(F)cc1-c1nc(-c2cccc(Cl)c2)nn1C1CCCOC1 Cn1cc(C(N2CCC(n3cc(Cn4cc(CO)nn4)nn3)CC2)=O)nc1O C(C1c2ccccc2CCN1c1ccncc1[N+](=O)[O-])NC(C(C(C)C)C)=O Cc1cc(N(C2CNCCC2(F)F)C(c2cc[n+]([O-])cc2)=O)n2nc(C)cc2n1 CCC(CC(C)C)C(=O)NCC(CCOC)NC(C1CC(SC)C1)=O c1(NC(CCN(C(C23COCC2C3)=O)CC)=O)ccc(C)cc1 CCCC(C)(O)C(=O)NCCNC(c1ccc(-c2ccc(CCF)cc2)cc1)=O CN1CCC(C(=O)N(C2CCCCC2)CCNC(c2cnc(S)nc2)=O)C1=O C1(NC(=O)C(F)CC2CCCCC2)CCC2CN(Cc3ccccc3)CC2C1 n1(C(C)C)cc(Br)c(C(=O)NCC2CCCCN2C(C2(C(N)=O)CCC2)=O)n1 C1(CN(C)C(c2cc[nH]c2C2CC2)=O)CN(C(c2cc[n+]([O-])cc2)=O)CC12CC2 Cc1nnc2n1CCC2(C)C(=O)NC1CN(C(c2csc(C#N)c2)=O)CC1C N1(C(C2(SC)CC2)=O)CC(C(=O)Nc2cccnc2OC(C)C)C2(CCC2)C1 N1(C(=O)CCc2ccoc2)CC2CCN(C(=O)Cc3ccc(F)cc3)C2C1 C(=O)(C(O)C(C)(C)C)NC(C1(O)CN(C(=O)CCCc2c(F)cccc2F)C1)C C1(C(N(CCC(=O)NCc2occc2C)CC)=O)CCC(N=[N+]=[N-])CC1 CC1c2cc(O)ccc2CCN1C(C1CCN(c2ncccn2)C1)=O Cc1nc(C(C)(C)C)sc1C(=O)NCC(C)N(C(=O)CCc1ncc[nH]1)C N1(C(CCOC(C)=O)=O)CCCN(C(C2CCc3n[nH]cc3C2)=O)CC1C(C)C CCCC(CC)N=c1[nH]c(=NC(C)c2nnc(C)o2)[nH]c2cc(OC)ccc12 c1(C(N2CC(O)(C(C)NC(C(C)=C3CCC3)=O)C2)=O)ncn2c(C)cc(C)nc12 C1(C(=O)NC2CC(C(C)O)C2)CCN(C(c2c[nH]ccc2=O)=O)C(C)(C)C1 n1(CCC)cc(CNC(C2CC(F)(CO)C2)=O)nn1 c1(OC)cc(C(=O)NC2CC2C(=O)Nc2ncco2)cc(Cl)n1 c1(C(=O)NCC(C)N(C)C(C2CC(CF)C2)=O)cccc(P(C)(C)=O)c1 c1(OC)cc(C(=O)N(C)CCN(C)C)c(NC(=O)Cc2cc(Br)ccc2F)cn1 CN1CCN(C(=O)CSCCC#N)CC1CNC(=O)C(O)CC1CCCC1 c1(C(N2CC(OC)C(NC(=O)C(C)c3ccsn3)C2)=O)cnn2c1CC(F)(F)C2 c1(C(=O)NC(C2CCCCC2)CNC(C2(O)CCCC2)=O)cc(C(F)F)ccn1 CP(C)(=O)C(CC(=O)NCC(CO)NC(=O)Cc1c[nH]ccc1=O)P(C)(C)=O CC1CCC2(CCN(C(=O)CN(C(=O)C3=NNC(=O)C3)C3CC3)C2)C1 CC(C)(C)C(=O)CCC(=O)NCc1cc(C(N2CC3CCC2C3)=O)cs1 CC(Cn1ccnc1)C(=O)NCC1(C(=O)N(C)Cc2ccoc2)CCCO1 c1(NC(C2CC(F)C2)=O)ccccc1CNCc1ncccn1 Cc1ccc(CNC(C2C(C)CN2C(=O)C=CCN2CCC2)=O)c(O)c1 C1(CNC(CC2(OC)CC2)=O)CN(C)CCN1C(c1cnc(C)nc1O)=O c1(C(=O)NC(C2(O)CCN(C(c3cc(C)sc3N)=O)C2)C)cncc2n[nH]cc12 N1(C(C23CC(C)(OCC2)C3)=O)CC2CCC1C1CN(C(C3CCS3(=O)=O)=O)CC21 N1(C(CCSC)=O)CC2CCC1C1CN(C(=O)CCc3ccc(Cl)c(F)c3)CC21 C1(CNC(C(C)CSc2ccccc2)=O)CN(C(=O)C(Cl)=CCl)CC1O C1(NC(C2(COC)C=CCN2C(=O)C=CC2CCCN2C)=O)CCC(=O)N(C)C1 N1(C(C(CSC)OC)=O)CCC2(CC1)CC2(CO)CNC(=O)COC1CCC1 c1(C(N2CCN(C(c3cscc3C(F)F)=O)C(CCO)C2)=O)cc(O)cc(=O)o1 N1(CCC#C)CCN(C(=O)C(C)C(C)NC(=O)CC2CCC(C)(C)O2)CC1 C(C(C)C(C)CC)NC(C1(CCC=C)CN(C(=O)CCCC#N)C1)=O C1(NC(c2cc(C)n(C)n2)=O)CC2CCC(C1)N2Cc1cc(C(F)(F)F)on1 CC1(C)CN(C(C23CCCCC2C3(F)F)=O)CCC1NC(=O)C1=CCOCC1 N1(C(C(c2ccncc2)C)=O)CC(C)(C)CC1CNC(=O)CC1CC1 Cc1ccn(C)c1C(=O)NC1CCN(C(=O)C=CC2CC2)C1Cc1ccccc1 Cc1cc(C(=O)NC(CC(=O)N2CC=CC2CF)C2CC2)nc(O)c1 c1(C(=O)OCC)cc(C(=O)O)[nH]c1C=Cc1cnc(C2CCOCC2)s1 C12(CNC(=O)Cc3nnc(O)s3)CCC1CCN2C(=O)CSC(F)(F)F C=C1CCN(C(=O)C(CC)CC=CC)C(C(=O)N(CC2=CCSC2)C)C1 c1(N(CCN(C(=O)C=Cc2cccc(Cl)c2)C)C)c(C#N)c(=O)n(C)c(=O)n1C N1(C(C(C)SC)=O)CCC(CF)(NC(=O)CCc2cnc(C3CCC3)o2)C1 CC1(CC(N2CC(CCCCNC(c3ccoc3Cl)=O)C2)=O)CCS(=O)(=O)N1 c1(OC)ncnc(C(=O)NC(C)C(C)(C)NC(=O)Cc2cnn(C(C)C)c2)c1F c1(C(=O)NC(C)CN(C(=O)CSc2nncn2C)C)cc(N=S(C)(C)=O)ccn1 C(=O)(C(CNC(=O)C(C)CC(=O)OCC)C(C)C)NC(CCOC)(C)C c1(C(=O)NCCC2(O)CN(C(C3CCCC(C)C3)=O)C2)cnn2c1CC(F)(F)C2 S(=O)(=O)(c1ccc(N2CCC3(C2)CC(F)(F)C3)cc1Cl)NC(c1ncc(C)o1)C C(=O)(C1=CCC(C)(C)CC1)N1CCC(C)(NC(c2ccc(C)o2)=O)C1 Cc1ncc(C(=O)NCC2(CC(=O)NC(C)C(C)CO)CC2)n1C Cc1cccc(C(N2CCCCC(CNC(=O)C(O)CC3CC3)C2)=O)c1C#N C12(C(=O)NCC(CNC(C(C)OC(C)(C)C)=O)F)CC3CC(C1)CC(C)(C3)C2 CCCCC(C)(c1nnnn1C)NCCc1cccc(Cl)c1 C1(NC(c2ccc(C(C)C)o2)=O)CN(C(C2CCSC2)=O)CCC1(C)C N1(C(c2c(C)nns2)=O)CCC(C)C(NC(C2(F)CCCCC2)=O)C1 c1(C(=O)OC)cccc(C(=O)N(CCCNC(=O)CC(C)F)C2CC2)n1 C(=O)(C(C)S(C)(=O)=O)NCC(CNC(=O)C)(C)C.c1(C(C)C)nncn1C1CC1 CN1CCCC1C1CCCN1C(=O)NC(CO)C1(O)CC1 C(CC(O)CNC(=O)CCc1nc(-c2ncccn2)no1)NC(C1C(OC)C1)=O C(=O)(CCC(=O)NCC1CCN(C(C23CC(C2)C(C(F)(F)F)O3)=O)C1)NC c1(C(=O)NCC2C3CN(C(CC4(OC)CCC4)=O)CC32)ccn2nnnc2c1 CN1CCCC(F)(C(=O)NCCCC2CCN(C(C3CCOCC3)=O)CC2)C1 c1(C(N(C(CN(C(c2ncc(CC)cn2)=O)C)C)C)=O)cc2ccc(C)cc2[nH]1 N1(C(CCC#N)=O)CC2CC2(NC(c2cn(CCc3ccccc3)nn2)=O)C1 C1(C(N2CC(C#N)(COC)C2)=O)CC2(CC2)CN1C(c1ccsc1C)=O c1(CCC(=O)NC(C(C)NC(C2(OC)CC2)=O)C)ccc(C#N)cc1F N1(C(c2cnc(CC)s2)=O)CCC(CO)(NC(=O)C(C)n2ccnn2)CC1 c1(N(C(c2c(OC)cc(OC)c(Cl)c2N)=O)C)ccc2c(c1)OC(F)(F)O2 C1(C(=O)NC(C)C=CC(=O)NCCC(C)C(F)F)(CC)CCOCC1 c1(NC(c2cn(C)c(=O)cn2)=O)c(-c2ccccc2)cc(F)cc1F Cc1nc(NCC(C)CNC(c2nc(C)n3c2CCCC3)=O)c(C)c(O)n1 N1(C(C(CCCC)=O)=O)CCC2(CCCCC2NC(=O)C=C2CCC2)C1 N1(C(C2C=C(C)CS2)=O)CCC(N(C)C(c2cc(C(F)F)no2)=O)C(C)C1 N1(C(C(=O)NC(C)C)=O)CC(NC(=O)Cc2cncs2)CC12CCCCC2 C1(CCNC(CNC(c2cc(OC)n[nH]2)=O)=O)CC2CCC1O2 C#CCC(C)C(=O)NC1CC(CNC(c2cnc(OC)cn2)=O)C1 N1(C(CC=CC)=O)CC(CNC(=O)C(C)COCC)C(F)(CO)C1 N1(C(C(=O)NC(c2noc(C)n2)CC)=O)CCC2(CC1)C(O)CC2O C=CCC(F)(F)C(=O)NCC1CN(C(c2ccc(NC)cc2)=O)C2CC12 c1(N(CC(=O)NC)C)[nH]c(=NC2CCC(C)(C)C(C)C2)nc2scnc12 c1(OC)c(C(=O)NC(CNC(C2(CO)CCCC2)=O)CO)cccc1F CC(C)(CC(F)F)C(=O)NC1CC2CCC1C(NC(=O)CCC1CC1(Cl)Cl)C2 N1(C(C2CCC(=C)CC2)=O)CCCCC(NC(C2CCCC(=O)N2C)=O)CC1 C1(O)(CC#C)CCN(C(C2COCCC2NC(C2(NC(C)C)CC2)=O)=O)CC1 C(=O)(C1CCCn2nccc21)NCC1N(C(c2c(C)ccnc2)=O)CCN(C)C1 c1(N(c2ccc(CN3CCC(C(C)NC(N)=O)CC3)cc2)C)cccc(F)c1Cl C(N=c1[nH]c2c(c(=NC(C)c3ncnn3C)[nH]1)CCCC2)C1C(CCC)C1 c1(C(=O)NC2CCN(C(C3(CC4CC4)CC3)=O)C2)ccc2ncnn2c1 N1(C(C2(C)CC3CC3C2)=O)CC2CCN(C(c3ccc(S(N)(=O)=O)o3)=O)CC2C1 Cc1cc(CCC(=O)NC(C)CC(C)NC(c2cnc(O)o2)=O)cc(C)c1 N1(C(C(C)=C2CC2)=O)CC2(CC(NC(c3c(C(C)C)cccc3F)=O)C2)C1 c1(NC(N(C(C#C)CC2CC2)CC)=O)c(OC)cc(OC)cc1C(N)=O c1(C(N)=O)ccc(Cl)c(C(=O)OCC2CCCC2C(F)(F)F)c1 C1(N(C(c2nccc(CC)c2)=O)C)CC2CCC(C1)N2C(=O)C(C)(C)F N1(C(C=CCCC)=O)CC(NC(c2ocnc2C(F)F)=O)CCC1C CC1(C#CC(=O)NCCNC(=O)CN2CC3CCC2C3)CCCO1 Cc1c(-c2nc(-c3ccc4c(c3)NCCC4)no2)cccc1[N+](=O)[O-] N1(C(C=CC(=O)OCC)=O)CCC(C(F)C(=O)NCC(C)CCO)C1 CCCCC(CNC(=O)C(C1CC1)C1CC1)NC(=O)Cn1cnc(C(N)=O)n1 N1(CC)CC(C(N2CCC(C)(NC(c3ncccc3Cl)=O)C2)=O)NC1=O C1(NC(c2ccsn2)=O)C2CC3C(C2)C13C(=O)NCC1(F)CC(CO)C1 C(CCC(=O)NCCCNC(c1cc(-c2ccc(Cl)s2)[nH]n1)=O)=CCC=C Cc1nc2ccccc2c(C)c1NC(=O)C(c1cccc(Br)c1)C N1(C(=O)OC)CCN(C(=O)C(Cc2cc[nH]n2)NC(C2C(C)C2C)=O)CC1 c1(C(=O)NCC(CO)NC(CC2(C#N)CCC2)=O)ccc2c(c1)NC(=O)CC2 N1(CC(=O)N(C(c2ccccc2)C)C)CCC2(CCC2)C(CO)C1 N1(C(c2ncc(OC(C)C)nc2)=O)CC2(C1)OCC1CC21 c1(OC)ccc(O)cc1C(N1CCC(C)(C(=O)Nc2cnc(C#N)nc2)C1)=O CC1OCCC1C(c1nnnn1C(C)(C)C)NCCC=CBr CCCC(C(=O)NC1CCC(CNC(C2(CC)COC2)=O)C1)c1ccc(Cl)cc1 C1(C(=O)NCC2(COC)CN(C(c3cccnc3S)=O)C2)CCC(=O)NC1 C12(NC(C(C)SC(C)C)=O)CCC1CN(C(=O)Cc1ccc(F)c(Cl)c1)C2 N1(C(C(C2CCC2)NC(c2c(C)n(C)cc2)=O)=O)CC2CC(C)C2C1 c1(NC(=O)NC2CN(S(=O)(=O)CC3CC3)CC2F)cc(Cl)cc(Cl)c1 CC(C(=O)NCC1(O)CCCN(C(=O)CCSc2ccc(F)cc2)C1)C(C)(F)F C1(C)(C(=O)NCCc2c(C)cncc2)CCCN(C(C2OCCCC2(C)C)=O)C1 C(=O)(CS(=O)CC)NCC(C)(C1CC1)NC(c1nc(CCCCC)sc1)=O c1(C(=O)NC2CC(NC(=O)CN(C3CC3)Cc3ccccn3)C2)cnncc1O Cn1c(NC(N2CCC3(CC2)COC(CO)C3)=O)nc2cccc(Br)c12 C1(CNC(=O)COC2CC=CC2)C(C2CC2)CCN1C(C1C2CCC1CC2)=O Cc1ccc(-c2ccnc(C(=O)CN(C)C)c2)cc1[N+](=O)[O-] Cc1cnc(NC2CCC3CC3CC2)c(S(=O)(=O)NC2CCC(C)CC2)c1 N12CC3(C1)CN(C3)C(=O)c1[nH]cc(c1)C2=O.C1(C(=O)OCC)(COC)CC1 c1(C(=O)NC2C(OC)CN(C(c3sc(N(C)C)nc3Cl)=O)C2)c(C)cccc1Cl C1(N(C)C(C2C=CCN(C(C3CC(O)CN3C)=O)C2)=O)CCOCC12CCC2 Cc1ccc(C(=O)NCCNC(=O)C(CC(C)C)N2CCCCC2=O)cc1CO C1(C(=O)NC2C(SC)CCC2)CC2CC1CN(C(=O)C=Cc1cocn1)C2 c1(C(=O)NC2CC3CN(C(Cc4n(C)nnc4)=O)CC32)cnc2n(c1=O)CCS2 C1(N(C(CC(c2cccc(OC)c2)C)=O)C)CCCCN(C(=O)CCC(C)C)C1 c1(C(N2C(CNC(C(C(C)C)n3cccc3)=O)CCC2)=O)cc2nccnc2[nH]1 C12(CNC(C=C(C)C(C)C)=O)CCCN(C(C3(Oc4ccccc4)CC3)=O)C1C2 c1(OC)cnc(C(N2CCC(CCN(C(=O)C(O)P(C)(C)=O)C)CC2)=O)c(F)c1 c1(CC)ccc(OCC(=O)NC2C=CC(CNC(=O)CCc3ccsc3)C2)cc1 C(C(C(C)C(C)C)NC(c1cnc(C)c(CC(C)C)c1)=O)NC(CCCC#C)=O O=C(N=c1ccn(Cc2ccc(F)cc2F)[nH]1)NC1CCN(CCO)C(=O)C1 c1(CC(=O)NCC2(F)CC(NC(c3csnc3Cl)=O)C2)ccc([N+](=O)[O-])cc1F CON(Cc1ccc(C)o1)C(=O)c1occc1CNC(=O)C(C)(C)O c1(C(N(CC(CC)NC(c2ccc(Cl)c(O)c2)=O)CC)=O)nn(C)c(C)c1Cl CSC1=C(C(=O)NCC(C)CNC(c2ccc(C)c(C#N)c2)=O)CCCC1 C1(C(=O)NCC(=O)NCC(=O)NC(c2cccnn2)C)CCC(=O)N1 C1(F)(C(N2CCC(O)(CNC(C(C)CN3CCOCC3)=O)C2)=O)CCN(C)CC1 Cc1cc(C(=O)NCC2CC(C)N(C(=O)C(C)CC3CCCC3)C2)c(N)c(Cl)c1 N1(CC(=O)NCC2(O)CCN(C(c3cccc(C4CC4)n3)=O)C2)CCNC(=O)C1 N1(C(C2C(C=C)OCC2)=O)CC2CCCC(CNC(c3nc(O)c(C)s3)=O)C2C1 C1(CC(c2ccccc2)C)CCCCN1N(C)C1CCC(C)(C)C1 C1(C(=O)NCc2ccc(Br)c(F)c2)CC2CCC1N(C(C1CCCS1)=O)C2 N1(C(C2CN(C)C(=O)CC2)=O)CC2(CCN(C(C3C4(CC4)C34CC4)=O)C2)C1 CN1CC(NC(=O)CC2(C)CCN2C(=O)C(F)CC2CCOC2)CC1CO C1(CCC)CCC(C(=O)NCCNC(=O)C(CC)N2CCCC2=O)CC1 c1(CN(C)C(C2(C(=O)O)CC2)=O)ncsc1C(F)(F)F Cc1nc(S(=O)(=O)NCCC2CCC(C)(C)CO2)c(-c2ccccc2)o1 c1(CNC(C(=O)N(CC(C)(C)N(C)C)C)=O)nc(C(C)C)ns1 c1(CC(=O)NCC(CNC(c2ccc(CCC)[nH]2)=O)CO)ccc(S(C)=O)cc1 N1(C(c2cc(C)n(-c3ccccc3)n2)=O)CC2CCC(CNC(=O)C(O)CF)(C2)C1 c1(C(=O)NC(CC)CNC(c2cc(C)nc(C(F)F)n2)=O)ccc(Cl)c(F)c1O c1(C(N(CC(CC)NC(=O)C(C)OC(C)=O)C)=O)ccccc1C(N)=O C(CC(O)C(C)C)NC(C1CC(CNC(C2(CC)CCOC2)=O)OC1)=O C1(CNC(c2n(CC)c(O)nc2)=O)(NC(=O)CN2CCOC2=O)CCCCC1C CCC(C)(C(=O)N1CCN(C(c2ncccn2)=O)CC(C)C1)C(N)=O c1(C(=O)NCC(C)NC(C(C2CCOCC2)OCC)=O)ncc(C)cc1Br C1(C(=O)NCCC2CCC(NC(c3cnn(C(C)C)n3)=O)C2)CCC2CC1CO2 N1(C(C2CCCN(C(c3cc(C)c(O)cc3)=O)C2)=O)CCC(F)(F)C(O)C1 N1(C(CC2(OC)CCCC2)=O)CCCN(C(=O)CC(O)CN(C)C)CC1C N1(C(=O)OC)CC2C=CC1C(C(=O)Nc1c(F)cccc1Cl)C2 C(=O)(C1=C(Cl)CCC(C)C1)NCC(C1CC1)NC(CCc1c(OC)cccc1)=O C(CN(C)C(C1CC1c1ccc(Cl)s1)=O)(CO)(CO)NC(C=CCC)=O C(=O)(N=c1cc(CC)n(C)[nH]1)C1CN(C(CC(C=C)(C)C)=O)CC12CCC2 CC1CCCC1(C(=O)NCCC1CC(O)C1)NC(c1ccccc1O)=O N1(C(c2cc(OC)c(F)cc2)=O)CC2CCC1C1CN(CCCC3CCC3)CC21 C1(SCc2nnc(C(=O)OCC)o2)Cc2cc(Br)ccc2O1 C(=O)(C1CCCn2cncc21)NCCC(C)CCNC(=O)COCCN(C)C N1(C(N(C)C)=O)CCCc2cc(NS(=O)(=O)c3cc(F)ccc3O)ccc21 N1(C(C(=O)N(C)C)=O)CCCC(CNC(C23COC(CCO2)C3)=O)CC1 c1(N2CC(CC(F)(F)Br)C2)ncccc1C(F)(F)F c1(OC)ncncc1NC(=O)CC1(C)CCN(C(=O)C(C)OC)C1 CC(C)C(O)C(C)C(=O)N1CCCC(CNC(c2cc(C(C)C)cnc2O)=O)C1 c1(CNC(=O)NCCCCS(C)=O)ccc(Br)cc1F CCC(CC(=O)N(CCCCCC(=O)NCC1CCN(C2CC2)C1)C)C(F)F C1(CCC=C)CCCN(C(CC2(C#N)CC2)C(=O)NC2(C)CC2)C1 C(C(C)(C)C1=CCCC1)NC(CCC1N(C(c2c(C)ccs2)=O)CCCC1)=O C12(C(=O)NCCCOC(C)C)COC(C1)C(NC(C1CCC1C)=O)C2 N1(C(C)=O)CC(C(=O)NCNC(=O)Cn2nc(C3CC3)ccc2=O)CC1(C)CO C#Cc1ccc(C2CC2C(=O)NC2CCN(C(c3cscn3)=O)CC2)cc1 c1(OCCC)cccnc1C(N1CC(NC(=O)CC2CCC(F)(F)C2)C1)=O N1(C(c2cnc(CC)nc2O)=O)CCCCCC(NC(c2cn(CC)nn2)=O)C1 N1(C(CCC=C(C)C)=O)CC2CS(=O)(=O)CC2(NC(=O)CCc2cc(C)no2)C1 N1(C(C2CC(C)(C)C2)=O)CCC(NC(=O)CC2(C)CC2(F)Cl)C(F)C1 C(=O)(CC(C)P(C)(C)=O)NC(CCC)CCCNC(=O)CS(=O)(=O)N(C)C Cc1ccc(-n2nc(C3CC3C)nc2C(C)CCN(C)C)cc1C S(=O)(=O)(CC1Cc2ccccc21)Cn1cc(-c2cccc(OCC)c2)nn1 c1(CN2C(C(N3CCCC(C(N(C)CC)=O)C3)=O)CCC2)ccc(O)cc1 C1(NC(C2N(C(C(C)C3CCC3)=O)CC(F)C2)=O)CC2C=CCC(C1)C2 N1(C(c2nc(C(C)(C)C)oc2)=O)CC2CC3CC2C1C3NC(=O)CC1CCCO1 C(=O)(CC(C)(C)C(C)=O)NC(CC)CCC(=O)NCC1(COC)CCC1 C1(NC(CS(CC)(=O)=O)=O)CC2CCCC(C1)N2Cc1cccc(CC(=O)O)c1 C(=O)(C1CCCc2c[nH]nc21)NCCCCNC(C=CSC)=O c1(CC(=O)NC2CCN(C(C3(C(C)(F)F)CC3)=O)CC2F)cccc2nonc12 Cc1c(C(=O)NCC2CC2NC(=O)C(CC(F)F)C2CC2)oc2c(C)cccc12 C(=O)(C1=CCCCO1)NC(CC(C)C)CNC(c1cncc(C(C)(F)F)c1)=O C1(OC)CCCN(C(=O)C(F)C2CC(NC(C3CC(C)(O)C3)=O)C2)C1 N1(C(C2(C#N)CCCC2)=O)CCC2(CC2C(=O)NCC2=NOCC2)C1 C(=O)(C(C)(C)C(C)O)N1CCC(C(C)NC(c2c(C)nc[nH]2)=O)CC1 c1(C(=O)NC2CN(C(CCNC(=O)NC)=O)C3C2C3)cc(N)cc(F)c1 Cc1cnsc1C(=O)N(CCC(C)NC(c1[nH]ccc1-c1cccs1)=O)C C1(c2ccno2)(C(=O)NCC(CO)NC(c2c(C)con2)=O)CCOCC1 C1(C(=O)NC(C#C)(C)C)CCN(C(c2cc3ccncc3[nH]2)=O)C12CCC2 C1(NC(=O)CNC(c2cccnc2)=O)CCN(C(c2ccsc2)=O)CC1CO C1(CC(=O)NCC2CCN2C(c2cc(O)no2)=O)COC(=O)C1 C1(C(=O)NCC(=C)CCNC(=O)Cc2nc[nH]n2)CCCCC1C(N)=O C1(CC(=O)NC(C=CC(=O)NCc2cc(COC)no2)C)CC(C2CC2)C1 N1(C(C(=O)NCC(CNC(c2cnc(COC)s2)=O)(C)O)C)CCCCC1=O Cn1ccc(C(N2CCN(C(C3CC(F)C3)=O)CC2)=O)cc1=O C1(O)(CNC(C2(C=C)CCC2)=O)CCCN(C(=O)C(F)(Cl)c2ccccc2)CC1 c1(COC)cccc(CC(=O)NCC(C)(CO)NC(C2(C)CCOCC2)=O)c1 CCCC(F)C(=O)NC(C)CC(=O)NCC(C)S(N)(=O)=O C1(NC(C2N(CC)CCC2)=O)CCCC12CN(C(C1SCC=C1C)=O)C2 Cn1cc(C(=O)NCC2(F)CCCN(C(=O)CN3CCC(O)CC3)C2)ncc1=O C(CC(C)(C)C(=O)NCC(O)(CO)CO)NC(C(C=C)C)=O C1(CC(N2CCC(C(C)(C)O)C2)=O)(NC(c2cc[nH]c(=N)n2)=O)CCCCC1 CCCC(CCCNC(c1cc(F)n[nH]1)=O)NC(=O)Cn1nccn1 N1(C(C(CC=CC)CC)=O)C2CCC1CN(C(=O)CCC(F)F)C2 C(=O)(C(F)(F)C1(O)CC1)NCC1C(NC(=O)C2CC2)C1 c1(OC)cccc2cc(C(=O)NCC(C)NC(C3CC(C)(C)CO3)=O)c(=O)oc12 C1(C)C(=O)NNC(=O)CN1CCO.Cc1ccsc1C(c1ccccn1)O N1(C(c2c(C)ocn2)=O)CCC2(CC1)CN(C(=O)CCCSC(C)(C)C)CCO2 C(=O)(C(C)CCCC(C)C)N1C(CN(C(=O)C(COC)CC)CC)CCCC1 Cc1cc(C(N2CCN(C(=O)C(C)CN(C)C)C(C(F)F)C2)=O)cnc1C C1(NC(CCC(C)C)=O)CN(C(C2COCCN2C)=O)CCC1O c1(C(=O)NC2CC(C)(NC(CC(C=C)CC)=O)C2)cccc2cnn(C)c12 C1(C(N(CC(O)CNC(C2C(C)(C)C2(C)C)=O)C)=O)Cc2nnsc2S1 N1(C(C(C=C)CC)=O)CCC2CN(C(=O)CN(C)C(C)C)CCC12 c1(C(N2CCC(CN(C(c3ccc(C)s3)=O)C)C2)=O)cnc(S)n1C Cc1cn(C2CCCCC2)[nH]c1=NC(=O)N(C1CCS(=O)(=O)CC1)C Cn1ncc([N+](=O)[O-])c1C(=O)NC1CCCCC1NC(c1cn[nH]c1)=O Cc1cnc(CC(N2CCC2CNC(=O)C(C2CCOCC2)O)=O)cn1 N1(C2CN(C(C)(C)CC3COC(C)(C)O3)C2)CCC2CC(C(N3CC(O)C3)=O)C2C1 c1(C(=O)NCCOCCCNC(COCCC=C)=O)ccn(CCF)n1 N1(C(CC(C)N(C)C)=O)CCOC2CN(C(=O)CSc3nnc(S)s3)CC12 C(=O)(C(C1CC1)N(CC(F)F)C)NCCSC c1(C(N2CC(CNC(C(OC)OC)=O)C3(C2)CC3)=O)ccc([N+](=O)[O-])nc1 N1(C(C2CCCN(CC)C2)=O)CCCCCC(NC(C2CC3CC2C3)=O)C1 N1(C(c2cc(COC)no2)=O)CCCCC1CC(N1CC(C(C)C)C1)=O C1(C(=O)NCC(C)NC(c2ccn3nccc3n2)=O)CN=C2N=CNN2C1 C1(CN(C)C(c2ccns2)=O)CCN(C(c2ccn(C(C)(C)C)c2)=O)C1 C(CCCC(CO)NC(C1CCCS1(=O)=O)=O)NC(CC(CC)OC)=O c1(CON=C(C(N2CCCC(COC)C2)=O)C)nccn2ccnc12 CC1(C)CC(C(=O)NCC2(F)CC(NC(c3ccc(Br)s3)=O)C2)C1 Cc1c(Br)ccc(NC(=O)NC(c2cc(Cl)cc(Br)c2)CO)c1F c1(C(N(C)CC2CN(C(=O)CSC3CC3)C2)=O)ccc(S(C)(=O)=O)cc1 C12CN(CC(C)(C)C1)C2=O.C1(NC(COC(CC)C)=O)(CC2CC2)CCC1 N1(C(COC(C)(C)C)=O)CCC2CN(C(c3sc(N(C)C)nc3Cl)=O)CCC2C1 C=C1COc2c(C(=O)NCC3CCN(C(=O)CCF)CC3(F)F)cnn2C1 Cc1cc(Br)cc2cc(CNCC(=O)OCc3ccccc3)[nH]c12 C1(C(N(C)CC2CCN(C(C3CC4C=CC3C4)=O)C2)=O)CCc2nnc(O)n2C1 n1(CC)cc(C(=O)NC(C2CCCN2C(C2CC(C)(C(=O)OC)C2)=O)C)c(C)n1 Cc1cc(CN(C)C)ccc1NCC12CC(C1)S(=O)(=O)C2 c1(C(=O)Nc2ccnnc2)cc2ccc(-c3cccc(F)c3C(F)(F)F)cc2[nH]1 C1(NC(C(CC)C)=O)CC12CCC(NC(c1c[nH]cc(Cl)c1=O)=O)CC2 c1(C(=O)NCC2CCC(NC(C3(C)ON=C(C)C3)=O)C2)cnc2c(c1)CCOC2 CCC(O)C(C)C(=O)N1CC(O)C(O)C1CNC(c1cc(CC2CC2)on1)=O C(=O)(CCC(N)CCC(=O)NCC1CC2CCC(C1)N2C(=O)C(F)(F)F)OC c1(C(=O)NCCN(C(=O)C(C)(C)C2CC2)CCC)cc(C)cc2c[nH]nc12 C12(C(=O)NCc3ccc(OC)cc3)C(NC(C3CC(F)C(=O)N3)=O)C3CC1C2C3 N1(C(CCOCCOCCC)=O)CC(C)(OCCC)C1.C(=O)(CCC1CC1)N Cc1nc2cc(C(=O)NC3CC4(C3)CC4NC(=O)COC3CCOC3)ccc2s1 c1(NC(C2C(C(=O)NCc3ccc(OCC#C)cc3)C2)=O)cc(Br)cc(C#N)c1 C1(CCC)COCCN1C(c1cnc(C)cn1)C(=O)NC1CC1 C1(C(N(C2(c3cc[nH]n3)CC2)C)=O)(NC(=O)COCc2nc[nH]n2)CC(O)C1 C1(CC(=O)NCC(C)(C)F)CCCN1C(C12CC(C(C)(C)C)(C1)C2)=O CC1=C(C)CC(C(N2CC(C3CC3C(=O)NCC3(C)CC(O)C3)C2)=O)CC1 C1(C(=O)NC2C(C)C2)CCC(O)CC1.c1(C(C)(C)C)cc(-c2noc(CO)n2)nn1C c12ncc(s1)C(=O)NCCCS2.c1(C(N2CC=CC2)C)nnnn1C1CCOC1 O=[N+]([O-])c1cc(F)ccc1CNC(=NCCCF)NCC1CC2CCC1CC2 c1(NC(C2(C#N)CC2)=O)cccc(NC(c2ccc(C(N)=O)[nH]2)=O)c1 c1(C(N(CC(CC)NC(=O)Cc2cccc(OC)c2Cl)CC)=O)ccc(N)c(N)n1 c1(CCC)cc(C(N2CC(NC(=O)Cc3cc(C)[nH]n3)C(C)C2)=O)c(C)o1 c1(C(=O)NCC(N(C(C2C(CC)CC2)=O)C)C2CC2)ccc(OC)nn1 c1(C(N2CCC(N(C)C(C3Cc4nncn4C3)=O)CC2)=O)cc2cccnc2s1 C1(NC(c2c(C)[nH]cc2)=O)CC12CC(NC(=O)CSc1nnc(S)s1)C2 c1(-c2cc(CNC(=O)NC3CCC(C(=O)OC)O3)no2)ccc(F)c(F)c1F N1(C(Cn2cnc(C#N)n2)=O)CC(CNC(=O)C=CBr)C2(CC2)C1 N1(C(CCNC(C)=O)=O)CC(O)(CN(C(=O)C2=CCC2)C)C1 C1(CNC(=O)CO)CN(C(C2CCN(CC(F)(F)F)C2)=O)CC12CCC2 C1(N(C(C=CCC)=O)C)CN(C(C2(COC)C=CCC2)=O)CCC1O C12CC(NC(=O)C(C(C)C)OC)(C1)C(C)O2.c1(OCC)ncc(C(=O)NC)s1 N=c1ccc(C(N2CC(NC(C3(Cl)CC3(F)F)=O)C(O)C2)=O)n[nH]1 C1(NC(Cc2c(C)non2)=O)CCC2CN(C(=O)CC3=NN(C)C(=O)C3)CC2C1 c1(C(=O)NCC2N(C(C(C=C)(C)O)=O)CC2)nn(C)c(C(F)(F)F)c1Cl N1(C(CCCC#C)=O)CC(C(C)(C)C)CC(CNC(C2(C)CCN(C)C2)=O)C1 CCCC(C(=O)NC1CC1NC(c1csc(C(F)(F)F)c1)=O)OCC N1(C(C2N(C(c3c(CC)occ3)=O)CC(C)C2)=O)CCC12CC(C)(CO)C2 Cc1nn(-c2ccccc2)c2sc(C(=O)NCC(C)N(C(=O)C(C)O)C)cc12 Cc1ccc(F)c(OCC(=O)NC(C)CN(C(=O)CC(C)O)C)c1 CC1C(NC(=O)C(CO)NC(C2CC2(C)C(F)F)=O)C1(C)C C#CC1(NC(=O)CC(C)CNC(C2(F)CCOC2)=O)CC(F)(F)C1 C(=O)(CCCN(C)N=O)NC1(C)CN(C(C2N(C(=O)OC)CSC2)=O)C1 N1(C(C2CCN(C(C)=O)C2)=O)CCC2CN(C(c3cccc(=O)o3)=O)C2C1 N1(CC)CCC(C(=O)NC2CC(CC(=O)NC3CCN(C4CCCCC4)C3)C2)C1 c1(CC(N2C(C(N(CC)Cc3ccccn3)=O)CC2)=O)cnccc1C CC1(C)C(=O)NCC1NC(c1ccc(Cl)cc1N1CCNC1=O)=O N1(C(Cn2nc(C)oc2=O)=O)CCCC(NC(C2C=CCC2)=O)CC1 Cc1c(C(N2CC(O)(CNC(C3CC4CC4C3)=O)C2)=O)sc(Cl)c1Cl N1(CCn2cc(-c3n(C)ncc3)nn2)CCN(C(=O)C(C)(C)OC(F)F)CC1 C1(CNC(C(C2(O)CCCCC2)CC)=O)(NC(C2(C(N)=O)CC2)=O)CCOCC1 C(=O)(C1=CS(=O)CCC1)N(C(C)CCNC(=O)COc1ccc(Cl)c(Cl)c1)C Cc1cc(CNC(C2CCC(CNC(C3(C)CCCOC3)=O)O2)=O)ccc1F C1(CC(=O)NC2(CNC(c3c(C)cc(C)o3)=O)CCCCC2)CCCCC12CC2 CN1CCOC(C(N2CCOC(CCNC(C3C4CC5C(C4=O)C35)=O)C2)=O)C1=O Cc1cnc(N2CCN(C(CO)CCC(C)C)CC2)nc1S(C)(=O)=O S(=O)(=O)(c1ccc(F)c2cnccc12)NC(C(=O)OCC)(C)C(C)C N1(C(CCC(=O)NCC)=O)CCC2CC2(C(=O)NCc2c(O)cccc2F)CC1 C1(C(=O)NC(CC#C)(C)C)CN(C(=O)CC(C)(C)O)CC1(C)C C1(CCNC(c2ccncc2F)=O)CCCN(C(C2CCCCC2O)=O)C1 c1(CNC(C2CCC(NC(c3[nH]cc(C)c3)=O)C2)=O)ccc(SC(F)(F)F)cc1 C(C)(C)(CC(F)C(=O)NCC1(CC)CCOC1)NC(c1cn(CCC)nn1)=O CN1CC2(CCN(Cc3ccc(C(=O)Nc4ncncc4Br)cc3)C2)C1 C1(N(C)C)(C(=O)NC2CC(NC(C34CC(CCO3)C4)=O)C2)CCCSC1 N1(C(C(C)(C)SC)=O)CC(CNC(C2COC(C)(C)CO2)=O)OC2(CCC2)C1 C1(C(=O)NCC(CNC(c2cnn(C)c2N)=O)F)CCc2nccn2CC1 N1(C(CC=CC=C)=O)CCCC(NC(c2ccc(C(F)F)c(OC)c2)=O)C1C C(CN=c1nc(N(C)Cc2cccn2C)c2[nH]ccc2[nH]1)C1CC(C)OCC1 CCCCC(C)C(=O)NC(C1(O)CN(C(=O)CCNC(=O)C(C)(C)C)C1)C C(=O)(CC(C)CN(C)C)N1CC(C(C)(C)O)(CNC(C2(C=C)CC2)=O)C1 c1(CC)ccc(C(=O)NCC(O)CCNC(C2(O)CCC2)=O)cc1Cl Clc1nc(Sc2ccc3ncsc3c2)c2sc(Br)cc2n1 CC(C)(CC#N)C(=O)N1CC(CNC(C2CC3C=CC2O3)=O)C(F)(F)C1 c1(C(=O)NCC(CC)NC(c2csc(NC(C)=O)n2)=O)ccc2nc(Cl)nn2c1 Cc1cc(N(C(=O)CC(CC2CC2)NC(=O)C(O)C2CCCC2)C)cc(C)c1 C1(CNC(c2c(CC)cco2)=O)CN(C(=O)CN2C(=O)CCC2=O)CC1O N1(C(CC(C)(C)C2CC2)=O)CC2CCCC1C2CNC(=O)C=Cc1nccs1 C1(CN(C)C(c2snc(Cl)c2Cl)=O)CCN(C(C2CCC3(C2)N=N3)=O)CC1 Cc1cc(C(=O)NC2CC(NC(c3occc3-c3ccccc3)=O)C2)cnc1O c1(OC)noc(C)c1C(=O)NCC1CCC(NC(=O)CCc2scnc2C)C1 N1(C(c2ccncn2)=O)CCC(O)(C(N2CCC(c3cccc(F)c3)C2)=O)C1 C1(CN(C(=O)C(C2CCN(C(c3csnn3)=O)C2)F)C)CCCC1(C)C C1(CNC(C2CCCN(C(C)C)C2)=O)CCN(C(c2cocn2)=O)CC1(F)F CCN=C(NCCCN1CCC1)NCc1ncnn1-c1ccccc1 Cc1nc(CO)ncc1C(N1CC(O)(C(C)NC(C2CCNC2=O)=O)C1)=O C(C(=O)N=S(C)(=O)c1ccnn1C)C1(NC(=O)OCC)CCC1 c1(OC(C(N2CCN(C(C3(CC=C)CC3)=O)CC2)=O)C(C)C)ccc(C)cc1C C1(C(N2CC(C)(OCC)C2)=O)CN(C(c2scc(C)c2C)=O)CC1(F)F c1(OCC(=O)NC2CC(NC(c3nc(C4CC4)cs3)=O)C(O)C2)cccc(Cl)c1 c1(C(N(CC(CNC(CS(CC)(=O)=O)=O)C)C)=O)cc(C)ccc1[N+](=O)[O-] C1(C(N2CCC(Oc3c(Br)cccc3Br)CC2)=O)CNC2(CC2)CO1 n1(CC(=O)NC2C(NC(C3(C(=O)OCC)CC3)=O)CC2)nnnc1C N12CC3CCN(C3C1)Cc1ccc(cc1O)C2=O.C1(CC)(CC)CCOCC1 Cc1nc(N2CCOC(C(C)NC(=O)CC34CCCN3CCC4)C2)ncc1Br C(=O)(C(O)C1=CCCCC1)N1CC2C(C(=O)NCC3(C)N(C)C(=O)CC3)(C2)C1 N1(C(=O)CCCF)CCC2(CO)CN(C(=O)Cc3cccc(Cl)c3)CC2C1 c1(N2CC(C)(CC(=O)NCc3c(O)cccc3O)C2)ncnn2cc(Br)cc12 C(C)(C)(CC(F)C(=O)NC(C1CCCCO1)C)NC(C(C)C(F)F)=O Cc1cc(=NC2CS(=O)(=O)CC2Oc2ccccc2)c2c([nH]1)CCC2 N1(C(C)=O)CS(=O)(=O)CC1C(=O)NCCOCCNC(C1CCCCO1)=O C1(N(C(C(CC)OCC)=O)CC)CCN(C(=O)C(C)N(CC(F)(F)F)C)CC1 c1(C(=O)NCC(c2ccccc2OCC(F)F)O)cccc(N2CCCC2)c1 c1(C(=O)OC)ccc(C(=O)NC2CN(C(c3nocc3Cl)=O)C2)cc1Cl c1(NC(C(c2ccn(C)c2)N(c2ccc(OCF)cc2)C)=O)ccc2c(c1)OCO2 c1(NC(C2C(NC(CC=CCC)=O)CCC2)=O)cc(Br)cc(C#N)c1 CC(CC(=O)NCC1(CNC(c2scnc2C2CC2)=O)CCOCC1)C(C)(C)C N1(C(c2c(C)cc(F)nc2)=O)CC2CC1CCC2NC(C1CN(C)CCO1)=O CC1=C(C(=O)NC(C2CCN(C(=O)Cc3ccnnc3O)C2)(C)C)CCCO1 c1(NC(C2CCC(CNC(=O)CC3CC(F)C3)O2)=O)ccc(F)c(C2CC2)c1 c1(OC)cccc(CCC(=O)NCC2CCC(NC(c3cncnc3C)=O)C2)n1 C(C)(CCCC(=O)N1CC(c2nncs2)C1)NC(C(=CC1CCCC1)C)=O c1(CNC(CC2(C)N(C(C3(C(C)=O)CC3)=O)CC2)=O)ccc2c(c1)CC2 Cn1ccc2c(C(=O)NCC3CC(F)CN3c3ncc(C#N)cc3Cl)cccc12 c1(CNC(C(C)OC(c2[nH]cc(C)n2)=O)=O)nc(O)c2ccccc2n1 CS(=O)(=O)c1ccc(C(=O)NC2CC(O)CN(C(c3ncc(Cl)cc3F)=O)C2)o1 C1(NC(C(C)SCCCC)=O)CCN(C(c2cn(C(C)(C)C)nn2)=O)CC1 N1(C(CCCn2c(C)nc(C)n2)=O)CCCOC(CCNC(C2(F)CC2)=O)C1 c1(CC(C)C(=O)NCC(C)(C)NC(c2nnc(S)n2C)=O)cccc(F)c1 CS(=O)(=O)C12COC(CNC3CCC3CCCl)(C1)C2 c1(C2CCN(C(C(=O)N(CC(C3CCCC3)C)C)=O)C2)ccccc1F C12(NC(=O)CCc3cn[nH]c3)CCCC1N(C(=O)CCC1CCCCC1)CC2 N1(C(C(CC)C)=O)CCC2OCCN(C(c3cc(C(F)(F)F)nn3C)=O)C2C1 n1(CCCC)ccc(C(=O)NC(C)(C)CCN(C)C(C2C=C(C)CS2)=O)n1 N1(C(C2CC(SC)C2)=O)CCC(C2CC2NC(C2CCCC3(CC3)C2)=O)CC1 C1(NC(COC2CN(C(C)=O)C2)=O)CC2CCC(C1)N2C(=O)CC1CCC2CC12 C1(NC(c2ccc(CNC(C3CC34CCC4)=O)s2)=O)CC2CCCCCC12 CCC(C)(CNC(=O)C(c1cccnc1)NC(=O)CC1COCCOC1)C(N)=O C1(CC)C(NC(=O)Cc2csc(C)n2)CCCN1C(=O)CC1CC1C(F)(F)F N1(CC2CC(OCC)C2)CCN(C(=O)CC2C(=O)NN=C2C)CC1C N1(C(C(CC)O)=O)CCC2(CC1)CN(C(C1CC=CCC1C(F)(F)F)=O)C2 C1(CCNC(CCSCC)=O)CN(C(=O)CC2CC(OC(C)(C)C)C2)CC1C N(C1CCc2cccc(COC(C)(C)C)c21)C(C1=NOC(C)C1)=O c1(N(CC(C)NC(=O)CCc2ccc(CO)cc2)C)cc(=O)n(C)c(O)n1 C1(CC)(NC(C2CCCC(N(C)C)C2)=O)CCN(C(=O)C=C2CCOCC2)CC1 C1(NC(CN(CCOC)C)=O)CN(C(c2c(C)cnn2C)=O)CCC1F c1(C(N2CC3(CN(C(c4ccc(Cl)cc4I)=O)C3)C2)=O)cccc([N+](=O)[O-])c1I CCCC(C(O)C(=O)NC(c1nc[nH]n1)C1CC1)NC(=O)C(C)N1CCCC1 C1(N(C(c2c(C)ocn2)=O)C)CCN(C(C2CC2CC(C)C)=O)CC1 CC1COCC(CNC(=O)C(C)(C)NC(=O)CCCOC(C)(C)C)O1 C=CCCCC(=O)NC(C1(O)CCCCC1)C(=O)NCC1CC(C)(O)C1 c1(NCCS(CCOC)(=O)=O)[nH]c(=NCCc2cnco2)nc2c1ncn2CC c1(N(c2ccc(OC)cc2)CCCNC(COC)=O)ncc2cn[nH]c2n1 C1(CCC(C)(C)NC(=O)COc2cccnc2)CCCCN1C(=O)C1=CCCS1 Cc1ccc(C)c(C(N2CC=CC(NC(=O)Cc3coc(C)n3)C2)=O)n1 O=C(C1=COCCO1)NC1CCCC(NC(c2cccc(OC(F)F)n2)=O)C1 CC(CC(=O)NC1(C)CN(C(C2CCC(C(N)=O)O2)=O)C1)C(F)(F)F CC(C)S(=O)(=O)CC(=O)NCC(O)CNC(c1cccc(OCCF)c1)=O C1(CNC(c2cc(C)ns2)=O)(CO)CCN(C(c2coc(C3CC3)n2)=O)C1 CC1CCC(C)(C(N2CC(NC(c3csc(-c4ccccn4)n3)=O)C2)=O)C1 c1(C(=O)NCC2CC(C)N(C(C3CC(C)(C(C)(C)C)C3)=O)C2)c[nH]c2ccccc12 c1(OC)ccc2oc(C(=O)NC3(Cc4cnn[nH]4)CCC3)c(C)c2c1 C1(c2ccccc2)(NC(C2C(CC)C2)=O)CC(NC(=O)Cc2c[nH]nc2O)C1 CCC(O)C(F)(F)C(=O)NCC1CC(F)(F)CN1C(C1CCC1(C)C)=O N1(C(Cc2n(C)c(S)nn2)=O)CC2CN(C(=O)CC3CCCCC3(F)F)CC2C1 C1(C(=O)NC(C(=O)N(C)C)CO)CCCCC1(C)NC(=O)C=CC(=O)NC1CC1 C(=O)(N=c1[nH]nc(Cl)cc1Br)C1CC(=C)CN1C(c1cccc(OC)c1O)=O c1(N2C3CC(C)CN(C3)C2=O)cc(Cl)c(O)c(Cl)c1.C12CCC(C1)C2(C)C.NC N1(C(c2c(OC)n[nH]c2)=O)CCC(CC(=O)NCC2OCCCC2(C)C)C1(C)C C1(NC(C(C=C)(C)O)=O)CC12CCN(C(=O)CCC(=O)N(C)C)CC2 N#Cc1ccc(C(N2CCCCC2CNC(=O)COc2ccc(CO)cc2)=O)o1 N1(C(CCNC(=O)NC)=O)CCC(NC(=O)CCc2nc[nH]n2)C(C(C)C)C1 CC(C)(O)C(F)C(=O)N1CC(NC(C2(CO)COC2)=O)C(c2ccc(F)cc2)C1 N1(C(CSCC)=O)CC(=O)N(Cc2nc(C3CC3)co2)C1=O N1(C(c2c(C)cccn2)=O)CC2(CCC2NC(c2ccccc2F)=O)C1 Cc1nc(Cl)ccc1CC(=O)N(C(CNC(C1(C)CC1(F)Cl)=O)C1CC1)C N1(C(C2C(=C)C2)=O)CCCC(C)(CNC(c2nc(C(F)(F)F)cs2)=O)C1 C(CC(C(C)C)NC(C1CCN(C(c2ccc(C#N)[nH]2)=O)C1)=O)OC CCCCC(O)C(=O)N1CC(C(=O)NCCNC(c2cnnn2C)=O)C1 C1(N(CC)CC2CC2)CCN(C2CC(CO)C(O)C2O)CC1 c1(SCC)cncc(C(N2CC(O)CC2CNC(c2sc(C)cc2OC)=O)=O)n1 N1(C(C(C)CC2CCC2)=O)CCOC(C(=O)NC2(C)CCC2)CC1 c1(C(=O)Nc2nccc(CN)c2)ccc(C2=CCCC2)cc1 c1(C(=O)NC(CCc2cccc(OC)c2)C(=O)O)c[nH]c2cncc(Br)c12 Cc1ccc2c(C(=O)NC34CCN(C(c5csc(Cl)c5)=O)CCC3C4)coc2c1 C1(C)(NC(Cc2cnc(C)s2)=O)CN(CC(=O)NC2CCC(C)CC2)CCO1 c1(CC(=O)N(C)C)ccc(C(c2ccccc2)N(c2scc(C)n2)C)nc1 C(CCCC(C)(F)F)(C(=O)NCc1nnn(C)n1)N(C1C(C2C(C)C2)C1)C c1(C(N2C(C(=O)Nc3cnc(C)nc3C)CCCC2)=O)cnn2ccccc12 N1(C(C2(SC)CCC2)=O)C2CCC1CN(C(c1cnn3ccccc13)=O)C2 C(CN=C(NCC(F)F)NC(C1(OC)CC1)C)c1ccc(OCC(=O)OC)cc1 CC1N(C(C2(C)CC(NC(c3sccc3C#N)=O)C2)=O)CCCC12CCC2 c1(CC)nn(C)c(Cl)c1C(=O)NCC1C=CCN1C(=O)C(C#N)CC c1(OCC)ccc(C(=O)NCCCCC(C)NC(C2(O)CCCC2)=O)cc1OC c1(C(=O)NCC(CNC(CNC(CC)=O)=O)C)cc(Br)cc(F)c1O c1(SC)nc(O)nc(C)c1C(=O)NC(C)CN(C(=O)CC1OCCO1)C N1(C(C)C)CCCC(CN2CC(Cc3ccncc3)C2)C1 N1(C(C(C2CC2)OCC)=O)CC(NC(=O)CCCF)CCC(O)C1 N1(C(C23CCC(CC)(CC2)OC3)=O)CC2=C(C1)CN(C(=O)Oc1ccccc1)C2 N1(C(c2sc(Cl)cc2Cl)C(=O)NCCCOC)CCCC2(C1)CC2(F)F N1(C(C(CC)C#N)=O)CCC(CNC(=O)CC2CCCOC2)(OC)CC1 CC1NC(=O)CCC1CNC(=O)C(N1CCCC(c2cccc(F)c2)C1)=O c1(C(N2CCC3(NC(c4ccn(C)c(=O)c4)=O)C(C2)C3)=O)cc2ccncc2s1 c1(N(CCCC)C2(c3ccccc3F)CC2)nccc(Br)n1 c1(C(=O)NC(C2CCCN(C(c3ccncc3F)=O)C2)C)ccc(F)c(F)c1Cl C(C(C(=O)NCCCSC(F)F)NC(=O)CCc1cnn[nH]1)OC C(=O)(C1=CC2CCC(C1)C2)N1CCC(N(C(CCSCCCC)=O)CCC)CC1 C1(C(C)NC(C2(C#N)CCCOC2)=O)CN(C(C2C3CC4C(C3)C24)=O)CCC1(C)C c1(C(=O)NC2CC(CCC(=O)NC3CCN(OC)CC3)C2)ccnc2cc[nH]c12 S(=O)(=O)(c1ccc(NC2CC(OCC)C2)cc1Br)N(C1CC(OC)C12CCC2)C c1(-n2cc(C3(NC(C4(C)CC4(F)Cl)=O)CCCOC3)nn2)ccc2ccccc2c1 c1(C(=O)NCCN(C(C(CCCC)NC(C)=O)=O)CC)onc2ccccc12 C1(C2N(C(CC=CC)=O)CCC2)CCCN(C(C2(CC=C)CCCCC2)=O)C1 N1(C(c2ccc(C)o2)=O)CCCC(C2CCN(C(C3(F)CCCOC3)=O)CC2)C1 N1(C(C2CN(S(CC)(=O)=O)C2)=O)CC(NC(=O)CC(C)C)CCC1C C12(NC(C3C(C)NCCC3)=O)CCC(CC1N)C2 c1(C(=O)NCC2C(NC(CC3(CSC)CC3)=O)C2)ccc([N+](=O)[O-])cc1Cl N1(C(C(C)Sc2nncn2C)=O)CC2CC(C1)C2NC(=O)C(F)(F)C(F)F c1(C(=O)NCC(O)CNC(c2cc(Cl)cs2)=O)cccc(CCCCO)c1 N1(C(c2nc(CC)sc2N)=O)CC(CNC(=O)CSCC(F)F)CC1(C)C C1(N(C(c2cc(C)nn2CC)C(=O)NCCC(=O)OCC)C)CC2CC1C1CC21 N1(CC(N2CCC(CC)C2CNC(=O)Cc2cncnc2)=O)OC(C)(C)CC1=O C1(C)(NC(CC=CC=C)=O)CCN(C(=O)COC(C)=O)C1 N1(C(c2c(CC)cc(N)cc2)=O)CCCC2CN(C(=O)COC3CC3)CCC12 C1(C(=O)NC(c2n[nH]c(=N)s2)C)COCCN(C(=O)C2=C(Cl)CC2)C1 c1(C(N2CCC(n3cc(C4C(C(=O)OC)C4C)nn3)C2)=O)cccnc1C(N)=O CCCC(C(=O)NC1CCCCC1CNC(=O)Cn1cnnc1O)c1ccccc1 C(=O)(C1CNc2ccccc21)N1C2CCC(CN(C(c3nc(C)oc3)=O)C2)C1 Cc1nc2cc(C(=O)NC(CNC(=O)Cn3cnnc3)CO)ccc2n(C)c1=O C(=O)(C(F)C(F)(F)F)N1CC(C(=O)NCCCC(C)(C)C)OCC1 C(=O)(C1=CCC(C)CC1)NC1(CC)CCCN(C(=O)COC(F)(F)C(F)(F)F)C1 n1(C(C)C)c(O)nc(NCC2(CNC(=O)CCCC(N)=O)CCC2)cc1=O c1(C(N2CCCC(=C)C2)C(=O)N(C2CCCCC2)CC)ncc(Br)cc1F C1(CNC(c2ccc(CSCCC)o2)=O)C(C2CC2)CCN1C(c1cn[nH]c1)=O Cc1cnccc1C(=O)NCC1CCC1NC(=O)CCOCC1CC1 C1(C(N(CC(C)N(C)C(c2cnc(O)n2C)=O)C)=O)CNC(=O)N1C c1(OC)sccc1C(=O)NC1COCC1NC(c1cnn(-c2cccnc2)c1)=O c1(C(N2C(C)CC(NC(C(C3CCCC3)OC)=O)C2)=O)cc(N)c(N)cc1F N1(C(C(CC#CC)NC(c2coc(C(C)C)n2)=O)=O)CCn2c(C)cnc2C1 c1(OC)ncc(C(N2CC(C(O)C(=O)NCCN(C3CCCC3)C)C2)=O)s1 C1(NC(CCCC(=C)C)=O)CC2(CCC(NC(=O)C(C)(C)CO)CC2)C1 C1(CC(=O)N(CCNC(=O)C(C2CC2)OC(C)=O)CC)CCC1(C)C CCC(O)CC(=O)NC12CC(C(=O)NC3CCCCC3F)(C1)C2 C#Cc1cccc(OCC(=O)NC2CC(N=[N+]=[N-])CN2)c1 N1(C(C(c2ccn(C)c2)C)=O)CCC(NC(c2cccc(F)c2)=O)C12CCC2 N1(C(CCCC(C)C)=O)CCC2(CC1)CC(C(=O)NCc1cc(=O)cco1)CO2 c1(NC(CC2(NC(c3cc(OC)c(O)cc3)=O)CCC2)=O)[nH]c(C)c(C)c1C#N C1(CC)OCCC1C(=O)N(CCNC(c1cnnn1C)=O)CCc1ccccc1 N1(C(c2c(C)ccs2)=O)CC2CCCC1C2CNC(=O)CCN1CCN(C)CC1 c1(C(N(C(CCNC(C2(OC)CCOC2)=O)C)C)=O)cn(C2CC2)c(C)cc1=O C(=O)(C(C)(O)CC)NCCN(C(=O)Cn1cc(C(F)(F)F)nn1)CC Cc1ccncc1-c1cn(CC2CCCN(C(=O)CCCc3ccsc3)C2)nn1 C(=O)(C(C)Cc1ccccn1)N(CC(CC)NC(=O)Cc1ncc(C)[nH]1)CC c1(CN2CC(NC(c3cccc(CCO)c3)=O)C(F)C2)cnc2n1CCOC2 c1(C(=O)NC2CC(F)(CNC(C(C)N(C(C)=O)C)=O)C2)n[nH]c2nccc(Cl)c12 CCC(CCOC)C(=O)NCCN(CC(C)O)C(c1coc(C)n1)=O CCC(CC)C(=O)NCC(CNC(C=CCN)=O)OC.C(C)=O N1(C(C2CC2(F)F)=O)CC2CN(C(C34CCCC3C4)=O)CC2C1 c1(C(=O)NC2CCC(C)(CNC(=O)CC3C=CCC3)CC2)cc(S(N)(=O)=O)co1 C1(NC(C(C)Oc2ccccc2)=O)CC2CCC(C1)N2C(C1CCCC12CC2)=O CC1N(C(C(=O)NCCOCC2CC2)C2CCC2)CCOC1(C)C c1(C(=O)NCC(CC=C)NC(=O)C(C)(O)C(C)C)ccc2[nH]ccc(=O)c2c1 C(C(CN=c1[nH]c(=NC(C)c2c[nH]ccc2=O)[nH]c2c1CCC2)OC)OC c1(C(=O)Nc2c(C(=O)NCCCCCN(C)C)nccc2)cc(O)c(O)c(O)c1 CC(C)C(CCNC(c1c(C2CC2)cnn1C)=O)NC(C1CCCS1)=O C(C)(C(CO)NC(=O)CSc1nncn1C)NC(C=CC(C)(C)SC)=O c1(C(c2nnnn2C2CCOC2)NC2(C=C)CCC2)ncc(Br)cc1OC N1(C(C2(OCC)CCC2)=O)CCCC(NC(=O)CN2CCC(=O)NC2=O)C(F)C1 C1(N(C(=O)C=CC2CCCC2)C)CC2CCC(C1)N2C(c1cc(N)cnc1Cl)=O C(=O)(C1=CC2C=CC1C2)NC1(CNC(C(CC(C)C)n2ccnc2)=O)CCCC1 c1(NC(CC(C)C)=O)cccc(NC(c2cc(-c3cccc(F)c3)no2)=O)c1C c1(C2C(=O)OC2)ccc(F)cc1.C1(N(CCOC)CCNC(C)=O)CCC1 c1(OC)ccc(C(N2CC3CC3(CNC(c3n[nH]c(C)c3O)=O)C2)=O)cc1O Cc1c(C(=O)NC23CC2CN(C(C2OCC2(C)C)=O)C3)cnc2ncnn12 Cc1c(CNC(C2CCCC(NC(c3cc(O)nc(O)n3)=O)C2)=O)cccc1O C1(OC)CC(NC(=O)OC(C)(C)C)CN(C(C2CCCCC2C(F)(F)F)=O)C1 c1(C(=O)Nc2cn(C)c(C(=O)Nc3cnccc3CO)c2)ccccc1C#N C1(NC(CC(=O)NC(C)C)=O)CN(C(c2cc(C(N)=O)c[nH]2)=O)C2(CCOC2)C1 N1(C(c2c(CC)nccn2)=O)CC(NC(c2c(Cl)nsc2Cl)=O)CCC(O)C1 N1(C(C)=O)CCCCC1CC(N1CC(F)CC1CN(C(=O)CC1CC1)C)=O c1(C2CCN(c3c(C(=O)OC)cncc3)C2)cccc2ccccc12 Cc1cc(=NCC2CC2C)[nH]c(NC(c2ccc3ncsc3c2)C)n1 c1(C(=O)NCC(CCNC(C2CC2F)=O)OC)cnnc(C)c1 c1(CC(N2CC3C(NC(C4CC(OC)C4)=O)C3C2)=O)cccc([N+](=O)[O-])c1 c1(C(N(C2CCCN(C(COCCN(C)C)=O)C2)CCO)=O)cc(=O)n(C)cn1 C1(C(N2CCN(CCNC(C3C(C)C3)=O)CC2)=O)COCCC1(F)F C(CCC(=O)NCCCC(C)NC(=O)C(C)OCC1CCCO1)NCC=C C(=O)(C(C)C(C)S(C)(=O)=O)N1CC(CNC(c2cn(CC)nc2C)=O)N(C)CC1 CCS(=O)(=O)c1cc(CNC(Cc2ccnc(Br)c2)COC)cc(Cl)c1 C(C(=O)NC1CC(C)(NC(C2(F)CCCC2)=O)C1)(C(C)C)NC(CC(C)C)=O N1(C(c2cnn(C)c2C#N)=O)CCCC(C2(NC(C3CC4(CSC4)C3)=O)CC2)C1 C12(NC(N(C3CC(CC)NCC3)C)=O)CCC(C(=O)OC)(CC1)C2 N1(C(c2ncc(C)nc2)=O)CC(C2CCCN(C(=O)C(C)(C)F)C2)C1 N1(C(CCCC(=O)NC(C)C)=O)CCC2(CC1)CC(NC(C1CC1F)=O)CCO2 C1(CC(=O)NCCC(C)O)CCCN(C(=O)COC2CCCC2)C1 C1(C(N2CCC(N(C(c3cncc(COC)c3)=O)C)CC2)=O)C2CCC(F)(F)C12 CCC(CC)CC(C(=O)NCCCF)N1CC(C2CC2)C1C1CC1 CCC(C)(C)CC(=O)N1CC(NC(c2cc(C)cc(C)c2)=O)CC(O)C1 C1(C(=O)NCc2cncc(C(=O)NC(C)CSC(F)F)c2)CCCCC(=O)N1 c1(CC)[nH]nc(C(N2CCC(F)(C(=O)NC(c3cn[nH]c3)C)C2)=O)c1C CC12C3C4C1C1C2C3C41C(=O)NC1CC(F)CN(C(C2CC2Cl)=O)C1 C=CCCC(C)(C)NC(c1cnc(CNC(c2ccc(CC#N)cc2)=O)nc1)=O c1(C(=O)NCC(CNC(C2C(C)(C)NC(=O)C2)=O)(C)O)cnc2[nH]ccc2n1 c1(OC)cc(NC(=O)C(C)(C)C2CCCN2C(=O)C(F)C(C)(C)O)ccc1O c1(CC)cc(CC(=O)NCC2(F)CCN(C(=O)C(C)CC)CC2)ccc1OCC c1(C(C)CC(N2CCC3C(NC(c4ccnc(S)c4)=O)C23)=O)ccc(F)c(F)c1 N1(C(c2n[nH]c3c2COCC3)=O)CCC2CCN(C(C3(O)COC3)=O)CC2C1 c1(CC)nn(C)cc1C(=O)NCC1C(C)CCN1C(=O)CCCC1CC1 Cc1cc(Cl)cc(C)c1OCCNC(c1nnnn1-c1ccccc1)C C1(CC=C)(NC(=O)COC2CCCOC2)CCN(C(=O)CSCCN(C)CC)C1 C#CCCCCCC(C(=O)NCC)N1CC(n2cc(C)cn2)C1 C1(C(=O)NC2C(C)N(c3nnc(O)s3)CCC2)CC2(CCCCC2)C1 CCCCC(CC(=O)N(C)CC1CCOC1)NC(c1cnn2cccc2c1)=O CCCCCCC(CC)C(=O)NC1CC(F)(CNC(c2c(C)nc(C)n2O)=O)C1 C12(CNC(COCC)=O)CCCC(CN1C(=O)CC1CCCCN1C)C2 C1(C)(C(=O)NCC2(C)N(C(c3nn(C)c(C(F)F)c3)=O)CCC2)CCCCCC1 N1(C(CNS(C)(=O)=O)=O)CCN(C(c2cccc(CO)c2)=O)CC(C)(F)C1 c1(NCC(C)C)cccc(C(F)(F)F)c1.c1(N(CC(C)C)C(=O)N)cccc(F)c1 C1(CC(=O)NCC2C(CNC(c3ccc(OCC)o3)=O)C2)CCCCC1(C)C C(CN=c1nc2sccc2c(NCC2CC2C2CC2)[nH]1)c1cncc(C)n1 C1(C(N(CC(=O)N(C)CCN(C)C)CCSC)=O)CCC(F)(F)CC1 N1(C(C(C)OCC(C)C)=O)CCCC(CC(=O)NC2CCCSC2)C1 c1(C(=O)NCC2C3CN(C(C4CC5(C)OCC4C5)=O)CC32)c(F)cc(F)cc1F c1(OC)cc(OC)c(CC(N2CCC(C(F)F)C2)=O)c(C(=O)O)c1 c1(NC(C2CC(CNC(c3cc(C)[nH]c3C)=O)C2)=O)ccc2n[nH]cc2c1 CCC(F)(F)C(=O)N1CC(NC(c2ccc(COC)nc2)=O)C(C)C1 C(C)(CNC(c1coc(C2CC2)n1)=O)(CO)NC(C1CC(SC)C1)=O c1(CNC(c2ccc(C(C)=O)[nH]2)=O)nc(C)c(C(=O)NCc2cocn2)o1 C(=O)(C1=C(C)CCCC1(C)C)N(C(C)CNC(=O)Cc1sc(C)nc1C)CC N1(C(C2(c3ccc(Cl)cc3)CC(N)C2)=O)CCCc2[nH]ccc2C1 c1(C(=O)NCCC(C(C)C)NC(CC2(C=C)CC2)=O)c[nH]c2nccc-2c1 c1(NC(=O)C(N2CCC3(CSC3)C2)c2nc(Br)cs2)ccc2c(c1)CCC2 N1(C(C(C2CC2)OCC)=O)CCCCCC1CNC(c1ccc(C)cc1CC)=O C12(CNC(CC3C(C)CCO3)=O)CCC(CC1)N(C(C1(C(F)F)CCCO1)=O)C2 C1(C(=O)NCCc2nnc(C)n2C)CC12CCN(C(=O)C#CC(=O)N(C)C)CC2 C(=O)(C(CNC(C1CC1F)=O)CC(C)C)NCc1c(C)cc(C)nc1 C1(O)(C(C)NC(=O)Cc2ccon2)CCN(C(=O)CCN2CCOC2=O)C1 c1(OCC)nccc(C(N2CC(NC(c3cncc(C(F)(F)F)c3)=O)C2)=O)c1F c1(C(N2C(C(C)NC(=O)CCC(N)=O)CCCC2)=O)cccc2c1CCC2 C(=O)(CCC#Cc1ccccc1)NC(C1(CNC(=O)C(O)c2ccco2)CC1)C C1(NC(c2c(CC)noc2)=O)CC2CN(C(c3cc(N)nc(Cl)c3)=O)CC2C1 C12(C(=O)Nc3c(CC)nccc3)COC(C1)C(NC(=O)CN(C)C1CC1)C2 N1(C(CC2(C)OCCO2)=O)CCC(C)(C)C(CNC(=O)CSC(F)(F)F)C1 Cc1ccc2c(C(=O)NCC3CC3CNC(=O)C(F)=CCCF)c[nH]c2c1 c1(C(N2CCC(C(=O)NCC3CC4(CCC4O)C3)(CO)C2)=O)coc2c1COC2 c1(SC)nc2ncnc(N3CC4C(CNC(C5COC(C)(C)C5)=O)C4C3)c2s1 N1(C(C(C)=C2CCCC2)=O)C(CC(N2CC(N(C)CCO)C2)=O)C2CCCC12 C1(C(NOCC(=O)OCC)=O)(CNC(=O)C(C)CO)CC(C)(C)C1 N1(C(C(C)n2cccn2)=O)CCS(=O)(=O)C(CCNC(C2(O)CCSCC2)=O)C1 Cc1cc(F)c(Cl)cc1C(=O)NC1CC(CNC(=O)C2=CCC2)C1 n1(CC)nnc(C)c1C(=O)NC(C1CCCCC1)CNC(C1CCS(=O)(=O)C1)=O C1(NC(c2ccoc2)=O)CN(C(c2coc(C3CCCC3)n2)=O)C2CC12 C1(N(C)C)CCCN(C(=O)C(C(C)(C)C)NC(c2cnn[nH]2)=O)CC1 C(=O)(N=c1cc[nH]cc1F)c1cccc(SCCc2c[nH]c(=N)s2)c1 c1(NC)cccc(C(=O)N(S(=O)(=O)CC2(OC)CNC2)Cc2ccccc2)n1 c1(C(=O)NCCCC(C)NC(=O)COC2CCCCCC2)cccc(F)c1C#N CC1(C)CN(C(C23CCCC2C3(F)F)=O)CCC1NC(C1CSCC(=O)N1)=O c1(C(N(C(CC(C)C)CO)Cc2c(F)cccc2F)=O)c(Cl)nc2ccccn12 c1(C(=O)NCC(C)(Cn2cccn2)NC(=O)CCOC2CCC2)ccc[n+]([O-])c1 CCC(CCCC(=O)NCCN(C)C1CC1)NC(=O)OC(C)(C)C C1(C2CCC2)(C(N(C(CNC(c2c(C)coc2C(C)C)=O)C2CC2)C)=O)CCC1 N12CCN1CC2C1CC1.c1(C=O)c(C2CC2)cccc1F.C=CC(O)C=O C1(NC(c2csnn2)=O)CC(NC(C2(c3cc(Br)ccn3)CC2)=O)C(O)C1 N1(C(Cc2ccc(C)nc2Cl)=O)CCC2(C1)CN(C(c1ccc[nH]1)=O)CC(C)O2 c1(C(=O)NC(C(N2CCC(OCC(=O)NC)C2)=O)c2ccco2)ccc(=N)[nH]n1 CC1(C)CN(C(=O)C(=O)NCC(F)F)CC1NCCCN1C(=O)CNC1=O c1(CNC2CCC(C(=O)Nc3cc(OC)c(O)cc3)C2)cccc2c1ccn2C C1(=CC(=O)N(C2CC(NC(c3ccnn3CCF)=O)C2)C)CC2CCC(C1)N2C N1(C(c2c(NCC)scn2)=O)CCOCC(CNC(=O)CC(C)CF)C1 N1(C(C=C(C)C(F)F)=O)CCN(C(c2cnn(CC3CCCC3)c2)=O)C2CC12 c1(C(N2CCCC(CO)C2)=O)ccc2c(c1)CN(c1ncc3ccsc3n1)C2 N1(C(C2(C)CC=CC2)=O)CC2CCC2(CCNC(=O)Cc2ccoc2)C1 Cc1nn(C)cc1CCC(=O)NC1CC1CNC(=O)Cc1nc[nH]n1 c1(C(c2cn(C)nn2)O)ccc2cc[nH]c2c1.Cc1nc2cc(n1)C1(CC1)N2 C1(NC(=O)CC2C=CC(NC(c3ccnc(S)c3)=O)C2)CCCC(F)(F)C1 Cc1ccc(Cl)c(C(=O)N(C(C)CCNC(=O)CC2CC3CCC2CC3)C)c1 c1(C(=O)NC(CC=C)CNC(=O)CC(F)(F)F)cc(-c2ccccc2)nc(O)c1 C(C)(CNC(c1cn(C)nn1)=O)(CC(C)C)NC(C(C1CCC1)OC)=O C(C)(CNC(=O)C=Cc1ncco1)(CC(C)C)NC(c1cc(CC)no1)=O N1(Cc2cc(C)no2)CCC(O)CC1C(=O)NCCc1ccccc1Cl c1(C(=O)NCC(CO)NC(C(CCOC)C)=O)cc(Br)c(F)cc1Cl C(CCCC(CO)NC(C1CC1c1nncn1C(C)C)=O)NC(COCC#C)=O c1(OC)ccc(COCC(C)C(=O)NCC(C2CCC2)NC(=O)C=C(C)Cl)cc1 O=C(CC1=CCCCC1)NC1CCSC12CN(C(C1CCc3cncn3C1)=O)C2 N1(C(c2c(CC)nns2)=O)CC(NC(C2CN(C(C)C)CCO2)=O)CC1(C)C N1(C(c2c(C)ncn2O)=O)CCN(C(=O)C(C)Sc2ccccn2)CC(C)(C)C1 Cc1n[nH]c(C)c1CC(C)C(=O)NCC1COCCN1C(=O)CCOC1COC1 CCCC(C(=O)NC1CC(O)(n2cc(-c3cnccc3Cl)nn2)C1)OC c1(OCCC(=O)OC)ccc(CNC(=O)N(CCCN2CCCCC2)C)c(C)c1 N1(CCC)CCCC1C(=O)NC1CCC(NC(=O)COCCSC)C1 C1(CC(=O)NC2CCCC2NC(C2CCCCO2)=O)CCCC1(F)F c1(NCCOC(C)C)ccc(S(=O)(=O)NCCC2CC=CCC2)cc1Cl Cc1c(Cl)cc(CNC(c2c(F)cccc2F)C2CCC2)cc1I N1(C(c2ccsc2)=O)CCOC2(CCN(C(c3nc(Cl)sc3Cl)=O)C2)C1 C1(N(C)C(c2cnon2)=O)CCCN(CCC2CCS(=O)(=O)C2)CC1 CC1(C)CN(C(C2(C#N)CCCO2)=O)CCC1NC(=O)CCCc1ccccn1 c1(NCC(CNC(c2cccc3c[nH]nc23)=O)O)ccc(Cl)cc1[N+](=O)[O-] Cc1cc(CC(N2CCN(C(c3cc(O)nc(Cl)c3)=O)C(CF)C2)=O)cc(F)c1 C(CCC(=O)N(CC(C)O)CCNC(=O)C(F)=C1CCC1)SC CC1(CNC(c2csc(C3CC3)n2)=O)CC(NC(=O)C(N2CCCC2)C2CC2)C1 C(CCCCC(=O)N1CCN(C(=O)CSCC(F)F)CC1CCO)NC(C)=O c1(C(=O)NC(C)CCCNC(=O)Cc2ccco2)coc2cc(F)ccc12 C1(NC(c2ccc(SC3CC3)cn2)=O)CCCC(NC(C2(C(=O)NC)CC2)=O)C1 C(=O)(C1=CCCOC1)NCCc1cc(C(N2CC(C(=O)OCC)C2)=O)no1 C1(C(N2CC(NC(=O)C=CC3CCCC3)C2)=O)(OC)CCCC1 CCCC(C)CC(=O)NC1COCCC1C(N1CC2CCC2(C)C1)=O C1(Cc2cn(Cc3cc(C)sc3)nn2)CCCCN1C(=O)Cc1sccc1C N1(C(C=Cc2occ(C)n2)=O)C(C)CC2CN(C(c3cncc(CO)c3)=O)CC12 Cc1c(C(N2CCC3(CC3NC(=O)C(C3CCCCC3)C)C2)=O)cccc1Cl Cc1nn(C)c(Cl)c1CC(=O)NC1CN(C(=O)C(O)CN2CCCC2)C1 c1(C(N(CCCn2cc(C3C4COCC34)nn2)C)=O)ccccc1C1CC1(F)F c1(CCCCC(=O)NC(C(CC)CC)C)cccc2ccc(C)nc12 [N-]=[N+]=NCC(C(=O)NCC1CC1Cl)NC(=O)Cn1cnc(=N)[nH]1 c1(C(N2CCCC(N(C(=O)CC3COCCO3)C)CC2)=O)cccc(P(C)(C)=O)n1 C1(C(=O)NCC(COCC)C)C2CC(O)C(C2)N1C(C1(C(=O)C2CC2)CC1)=O C1(C(=O)NCc2c(C(=O)NCc3cnc(C)s3)occ2)CCC(O)CN1C c1(C(=O)NC2CCN(C(c3[nH]cc(CC)c3)=O)CC2C)cccc2cc[nH]c12 C1(NC(C2CC2[N+](=O)[O-])=O)CCC12CCN(C(c1cc[nH]c3nccc1-3)=O)CC2 Cc1cc(C(N2CC(C(N)=O)(CNC(C3(C)CCCC3O)=O)C2)=O)nn1C CCC(CC(F)F)C(=O)N1CCCC(CC)(NC(c2sccc2Cl)=O)C1 c1(OC)ccc(CC(C2CC2)N)cc1.C1(=O)CC(CF)NC1=O.C(C)(C)(C)O N1(C(CN(C)C)=O)CCC(n2ccc(NC(=O)Cn3cncn3)n2)CC1 N#Cc1ccc(C(N2CC3(CC(C(=O)NCc4sccc4Cl)C3)C2)=O)c(F)c1F N12CCc3cc(ccc3C1)C2=O.c1(C(C2CCC2)C)ccc(F)c(C(F)(F)F)c1 N1(C(c2cncc(C(=C)C)c2)=O)CCN(C(=O)CC2CC(=C)C2)CC12CCC2 C(=O)(C(CCOCCO)NC(=O)C=CC(C)(C)SC)N(C(C=C)C)C C1(CNC(CC2(N(C)C)CCC2)=O)CN(C(c2cncn2C)=O)C2CCCC2O1 Cc1ccccc1C(CNC(=O)C(C)NC=O)NCCC(C)C c1(C(=O)NC2C3N(C(C4(CC=C)CC4)=O)CC(CC3)C2)cc2cccc(F)c2o1 C1(NC(C2CCCC(O)C2)=O)CC2(CCCCN2C(=O)Cc2ncc(Cl)s2)C1 CC(C)CC(N=c1[nH]c(C2CC2)nc(=N)[nH]1)C1CC1 c1(OC)ccc(-n2nc(-c3nc(C)cs3)nc2C2CN3CCN2CC3)c(C)c1 C1(C(c2nnnn2C2CC2)NCC2(C#C)CCC2)(C(=O)OCC)CC=CCC1 C1(NC(c2c(C)cccc2Cl)=O)CCC2(C1)CN(C(=O)C(C)O)C2 c1(CC(=O)NCCCNC(C(C)n2cccn2)=O)ccc(Cl)cc1Cl N1(C(c2c(CC)csc2)=O)CCCC(CNC(=O)CC(c2ccccc2C)C)C1 C12(CNC(CC(C)(C)OC)=O)CCC(CN(C(c3ccnc(C)c3C)=O)C1)C2 c1(NC(=O)C(=O)NCC2CCN(CC)C2)ncnc(C(F)F)c1Br Nc1ccc(F)c(F)c1C(N1CC(NC(C2CC(=O)NC(=O)N2)=O)C(F)C1)=O Cc1ccc2oc(C(N3CC=CC3Cn3cc(C4(C)CCCO4)nn3)=O)cc2n1 CC1CN(C(=O)C(=O)NCC2CC2)CC2(CCN(C(C3CCCC(=O)C3)=O)C2)O1 C12(NC(C=CS(CC)(=O)=O)=O)CC(CNC(C3CCCC3)=O)(C1)OC21CCC1 n1(CC(=O)NC(CNC(c2csc(C)c2C)=O)(C)C2CCC2)nc(O)ccc1=O N1(C(CC=C(C)C)=O)CCCC2C1CCCCN2C(=O)C(N1CCCC(C)C1)=O c1(CNC(C(c2ncccc2F)N2C(CCCC)CCC2)=O)cccc(C)c1 C1(NC(c2c(C)c[nH]n2)=O)CN(C(=O)CN(C)C(=O)C2CC2)C(C)(C)C1 N1(CC(=O)NC(C(=O)N(c2ccccc2)C)CCC2CC2)CCc2ccsc2C1 N1(C(C(C)C2CC2)=O)CCC(CF)(NC(C2CCN(C3CCSC3)CC2)=O)C1 N1(C(c2c(CC(=O)OC)occ2)=O)CCN(C(=O)CNC(=O)C(SC)SC)CC1 c1(NCC(CC)n2cccn2)ncc(C)cc1S(=O)(=O)NC1(CC)CCCCC1 C(C1=CCSC1)(c1n(C(CC)C)nnn1)NCc1nccn1C(C)C Cc1coc(C(=O)NC2CC(NC(C3(CCN(C)C)CC3)=O)C2)c1C c1(C(=O)OC)cncc(-c2cn(C(C)C(N3CC(O)CC3C)=O)nn2)c1 N1(C(c2ccc(F)c(O)c2)=O)CCC2(CC1)CN(C(C1CCSC1)=O)CCO2 C(CN=c1[nH]cncc1I)(C(C)(C)C)NC(c1ccn(CCOC)n1)=O C1(NC(c2c(COC)ncs2)=O)CC(F)CN(C(c2cnoc2C)=O)C1 N1(C(C(CC(C)(C)C)O)=O)CCC2CCC(C1)N2C(c1ccn2nccc2n1)=O C(=O)(C(C)P(C)(C)=O)N(C(C)C)CCNC(=O)CC1CCNC(=O)C1 N1(C(=O)NCC(C)N(c2ccccc2)C)CCOc2cc(CN)ccc2C1 C1(C(=O)NC2COCCC2NC(C2(CC3CCC3)CC2)=O)CCC(F)(F)CO1 C1(NC(c2cnnn2C2CC2)=O)CN(C(c2cccc(F)c2O)=O)CC1C1CC1 C1(OC)CCC(C(=O)NCC(C(=O)N(C2CCOC2)CCO)N(C)C)C1 CCNC(=O)COC(F)F.C(C(C)C)SCCCCSCCCl c1(C(c2nnnn2CCC2(C)CC2)NCC2(CCOCC)CCC2)ncsc1Br C1(C2(NC(=O)CCNC(c3cc(C)c(C)s3)=O)CC2)(OC)CCC1 C1(NC(C2CCCN(C(C(C)(C)N=[N+]=[N-])=O)C2)=O)C2CCCC1COC2 CC12CCOC(CNc3cc(OC4CCNCC4)ccn3)(C1)C2 Cc1cnc(C(=O)NCc2ccc(CNC(C3(C)CCNC3=O)=O)cc2)cc1Cl C=C(Cl)CC(C(=O)NCCC1(O)CCCC1)NC(=O)C(N)=O N1(C(C2CCCSC2)=O)C2CCC1CC(NC(C1(Cl)CC1)=O)C2 C=C1CCN(CC(=O)Nc2scnc2-c2ccccc2)C(C(=O)OC)C1 C1(C(=O)NCC(=C)F)CC(NC(=O)CCCF)C12CCC2 CCC(C(=O)NCC(C(C)(C)C)NC(=O)COCCSC)C(F)(F)F C(=O)(C1=CCCCC1)N(CC1(C)CCN(CC2(c3ccc(F)cc3)CC2)C1)CCl C=C=CCCC(=O)N1CCC(C(=O)NCC2(F)CCN(C)C2)(CC)C1 C(=O)(CCCCC(=O)NCC(C)(C)CCNC(c1nccc(Cl)c1F)=O)OC C(CCC)(C(=O)NCC12CC1CN(C(C1(COC)COC1)=O)C2)=CCC C12(C(N3CC=C(CNC(CCc4ccc(C)s4)=O)CC3)=O)CCCCC1C2(F)F C1(NC(CCN2CCN(C)CC2)=O)CCCN(C(C2CCCC(F)(F)C2)=O)CC1 c1(C(N2CC(F)(CNC(C3(COC)CC3)=O)C2)=O)cc(=O)n(C)cn1 Cc1cc(C(=O)NC2CC3CC2N(C(c2ncc(N)cc2C)=O)C3)cc(C)c1F N1(C(C(=O)NCCOCC)=O)CC(NC(=O)CCOC(C)=O)CC(F)(F)C1 c1(-n2c(C3CC=CC3)nc(C3CCOC3)n2)cccc2cnccc12 C1(C(=O)Nc2c(CC)noc2)CC2CC1CN(C(=O)C1=CCCCC1C)C2 C(=O)(C(C(C)(C)C)N(C)C)N1C(C)(CC(=O)N(C(C)CO)C2CC2)CC1 c1(C(=O)NC(C(c2ccccc2)NC(CCC2C(C)C2)=O)C)cc(C#N)no1 C=CCC(C)C(=O)N1CC=CC(N(C)C(c2ccc(C(N)=O)[nH]2)=O)C1 C12(COC)CN(C(C3CC4CCC(C3)C4)=O)C(CNC(=O)C(C)OC)(C1)C2 C(=O)(C1=CCCS1)N(C(C)C)CCNC(=O)CC1CC1C(F)(F)F c1(C(=O)NCCCOCCNC(C2(CC)CCCC2O)=O)cccc(F)c1F C1(NC(c2ncc(C)nc2)=O)CN(C(=O)COC2CC2)CC1S(C)(=O)=O CCCCC(CNC(=O)C=CC(C)(C)C)NC(=O)CNC(=O)Oc1ccccc1 c1(CNC(CN(CCC)C(c2c[nH]nc2Cl)=O)=O)nocc1C(C)C C1(C(N2CCC(C)(NC(C3C(CCOC)C3)=O)CC2)=O)CCC2(CCC2)OC1 N1(C(=O)NCC(C2CCCCC2)C)CCOCCC12CCOCC2 C1(CCNC(C=CCCC)=O)CCN(C(c2nc(OC)ccc2F)=O)C(C)C1 N1(C(CN(C)CC)=O)CC(NC(=O)C(c2ccc(C)cc2)C)CC(F)C1 c1(C(N2CCC(O)(C(C)NC(=O)CS(C)(=O)=O)C2)=O)cn(C)c(=O)nc1O C(c1ccc(C2CC2)cc1)=CC(=O)NC(CN(C(CCC(C)OCC)=O)C)C C1(COC)(CNC(=O)C(C)OC2CCCC2)CCCN1C(c1coc(CO)c1)=O C(=O)(C(C)(CO)NC(=O)C(=O)C1CCCC1)NC(CC(=O)OC)C C1(CNC(CP(C)(C)=O)=O)CCCCCN1C(=O)CC1(O)CCOCC1 n1(CC)ccc(C(=O)NC2CCCC2NC(=O)Cc2nc(C(C)C)c(C)s2)c1C CN1CCOc2c(C(=O)NC3CCN(C(C4CCC5(CCC5)C4)=O)C3)cccc21 N1(C(c2ccc(CSC)cc2)=O)CCN(C(c2[nH]ncc2C#N)=O)CC1C1CC1 c1(C(=O)NC(COC)CNC(C2C=CCC2)=O)ccncc1 c1(C(=O)NCC2CCOC2)nn2ccccc2c1C(=O)NCc1cn[nH]c1 c1(CC(=O)NCCOCCC(=O)NCC(CC)N2CCCC2)ccc(O)cn1 C1(C(=O)NC2(C(=O)OCC)CC2)CN(C(C2CC3C=CC2CC3)=O)C2(CCC2)C1 CCCCC(C)CCC(C)NCc1ccc(C)c(C(C)=O)c1 C1(NC(c2coc(Br)c2)=O)CC1C1CCCN(C(=O)COCC(F)(F)F)C1 Cc1nc2ccc(C(N3CC4CCC3C(NC(=O)CC=C(Cl)Cl)C4)=O)cc2[nH]1 C(=O)(CC(C(=C)C)OCC)N(C1CCN(C(C2CC(=C)C2)=O)CC1)CC N1(C(Cc2cnc(C)[nH]2)=O)CCN(C(=O)CCOCC(N)=O)C(CC(=O)NC)C1 c1(C(N(CC(=O)NC)C)=O)ccc(CNCCNS(C)(=O)=O)cc1 C#CCC(CC(=O)NC1CC(CC(C)(C)C)C1)NC(=O)CC1CCCNC1=O C1(CNC(c2sccc2F)=O)CN(C(=O)CC2CC=CCC2)CC1C(F)(F)F C(C(C)(CO)CN=c1cc(C)nc(N2CCOCC2)[nH]1)OC.C1(C(C)(C)C)CN1 Cc1ccc(C(C)CC(=O)NC2CC(C)(NC(C3CCNC(=O)C3)=O)C2)cc1 C(=O)(C(C)(C)CO)N(CCNC(C(n1ccc(C(F)(F)F)n1)C)=O)C CCC(C)CC(=O)N1CCC(C)C1CNC(C1(COC)C=CCC1)=O C(=O)(C#CC1CCOC1)NCCCNC(C(c1ccc(C#N)cc1)O)=O Cc1nc(N2CCC3(CCC(C)C3)C2)nc2c1NC(=O)C(C)N2C C1(C(=O)NCc2ncc(C)nc2)CC2CCC1N2C(c1nnn(C)c1N)=O O=C(CN=c1[nH]c(=NC2CCS(=O)CC2)[nH]c2ccccc12)NC1CC1 c1(OCCC)cccc(C(=O)NC2CCCCC2CNC(C2SCCCS2)=O)c1 CC(C)(CC(F)(F)F)C(=O)NCC1CCCN1C(C1CCCN1c1nccs1)=O c1(CN(c2cc(Cl)sc2C)C(CN(C(COC)C)C)=O)ccccc1C C(CC(O)C(=O)N(C1CCCC1)CCNC(=O)C(F)(F)CN(C)C)N(C)C c1(CC(=O)N(C2CCCN(C(=O)CCCc3cccnc3)C2)C)c[nH]ccc1=O C1(C(=O)OC)CCN(C(=O)CC2(C)CCN2C(=O)C(C)CSC)C1C N1(C(C2(OC)CCCOC2)=O)CC2(C1)CN(C(=O)CC(C)C)CC(C)(C)O2 CCC(C)(CO)C(=O)NCC1CC(F)CN1C(C1CCC(=O)N1C1CC1)=O C(CCC(N)C(=O)NCc1ccc(Cl)c(NS(C)(=O)=O)c1)OC [N-]=[N+]=NCCCC(=O)NC1CC(F)CN(C(=O)CS(N)(=O)=O)C1 CC1=C(C(=O)N2CC3CCC2C(CNC(=O)CCc2nc(O)n[nH]2)C3)SCCO1 c1(SC)nc(NCC23CC2CN(S(=O)(=O)Cc2ccc(Cl)cc2)C3)ncc1F N1(C(C(C(C)C)O)=O)CCC(CNC(=O)CC(C)(O)C(F)(F)F)C(F)(F)CC1 C(=O)(C1c2c[nH]nc2CCC1C)NC1(C)CN(C(C(CC=C)(F)F)=O)C1 C(=O)(CC(C(F)(F)F)NC(=O)CC1CCCSC1)N(C1CC(O)C1)C c1(OCC)nc(N2CCC(NC(c3cc(O)nn3C)=O)C2C)ncc1Cl C12(CNC(c3ccccc3C3CC3)=O)CCCC1CCN2C(=O)CC1CCC1 c1(C(C)C(=O)NCC2CC2NC(=O)C(N2CCSCC2)C)ccc(-c2ccccc2)[nH]1 C1(C(=O)NC(c2ccccc2)C(=O)Nc2cn(CC=C)nc2)CC(=O)NC1(C)C C1(C2CCN(C(C3COCC3(C)C)=O)CC2)(NC(c2[nH]c(=NCC)sc2)=O)CC1 N(C1COc2ccc(F)cc21)c1cc(NCc2ccc(C#N)s2)nc(C)n1 c1(CC)ncc(C(C(=O)NCCCC2CC2)N(C)CC2(C)CCCO2)[nH]1 Cc1cc(C(=O)NC2CCC(C(F)(F)F)NC2=O)cc(C)c1Br CC1(C)CN(C(=O)CSCCC#N)CC(CNC(C2Cc3ccccc3O2)=O)O1 C12(NC(CCOC)=O)CC3CC(C1)CC(CNC(C1COC4CC1C4)=O)(C3)C2 C1(C(=O)NCC2(COC)CN(C(=O)CCn3cnnn3)C2)CC12CCOCC2 c12ccc3c(c1)CN(CC3)C2=O.c1(CNC)cnc2c(C#N)cnn2c1 C1(CNC(C(C2CC2)OCC)=O)CN(C(C2(CN(C)C)CCCCC2)=O)CC1C C1(C(=O)NCC(O)CCNC(=O)CCC2CC2C)(OCC)CCSCC1 N1(C(C2N(C(CC)=O)CSC2)=O)CCN(C(c2cnc(OC)nc2)=O)C(C)C1C N1(C(c2n(CC#N)ncc2)=O)CC(NC(=O)Cc2ccnc(O)c2)C(C2CC2)C1 N1(C(c2nc(CC)sc2N)=O)C2CCC1C(NC(=O)CCN1CCCCCC1)C2 C1(OC)CCCN(C(=O)C(Cn2cccn2)NC(=O)C(c2ccn(C)c2)C)CC1 N(C(=NCCC(O)C(F)(F)F)NCc1cccc(F)c1)C(C=C)C c1(COC)nc(NCCC(N)=O)cc(=NCC(C)(C)c2c(F)cccc2F)[nH]1 N1(C(C(C(C)C)SC)=O)CCN(C(=O)Cc2nc(=N)[nH][nH]2)CC1C1CC1 N1(C(C2CCN(C(=O)NC)CC2)=O)CC(C2(NC(c3ncc(F)cn3)=O)CC2)C1 C1(NC(=O)Cn2cc(CN3CCCC3=O)nn2)CCC12CCCC2 N1(CC)CCN(C(=O)C(CO)NC(c2ccc(F)cn2)=O)CC1C c1(C(N(C2CN(C(=O)CCc3nncs3)CC2F)C)=O)cccc2nsnc12 Cc1cc(O)ccc1C(=O)NCC1(C(=O)Nc2cncc(CO)c2)CC1 N1(C(C(CC)=CCCC)=O)CCC(C(=O)NCC2CCC2CO)(OC)C1 C12(NC(COC(C)=O)=O)CCC(NC(=O)C(C)NC(c3ccco3)=O)(CC1)C2 c1(C(=O)OC)cccc(CN2CCC(c3cccc(Br)c3)C2)c1Cl C=CCCCC(C(=O)NC1CC2(CCC2)C1OC)NC(c1ccc(C)[nH]1)=O C1(C)(NC(c2ccc(Cl)c(F)c2)C)CCCN(c2cc(C(F)F)ncn2)C1 N1(C(C(F)=CCC)=O)CC(NC(=O)COCC2CC2)C(C2CC2)C1 C1(C(=O)NCCCCN(C)C)COCCN1C(C1CCCCN1C)=O C1(NC(C(n2ncc(C)c2)C)=O)CCCN(C(=O)CCCCc2cnn[nH]2)C1 C1(CNC(=O)C(O)CC(F)F)CC12CCN(C(c1ccc(F)c(O)c1F)=O)CC2 c1(CC)nocc1C(=O)NCCN(CC(C)O)C(c1nnc(C(C)(C)C)s1)=O c1(C(N2C(C3CCN(C(C4CCC(CC)O4)=O)C3)CCC2)=O)cn(C)c(=O)n1C CC(Cc1ccnn1C)C(=O)NC1CC(CNC(C2CNC(=O)N2)=O)C1 c1(COC)cccc(C(N2CCCCC2CF)C(=O)NCCCOCC2CC2)c1 c1(CNC(C(C)(C)C2CCCO2)=O)cccc(NC(=O)CCNS(C)(=O)=O)c1 CCC(C)CCC(=O)N1CC(NC(=O)Cn2cnc([N+](=O)[O-])n2)CCC1C N1(C(C(C(CC)(C)C)O)=O)CCc2nnc(N3CCCC3)cc2C1 n1(C(C)C)ncc(C(=O)NCC(C2CC2)NC(C2(CO)COC2)=O)n1 C1(C(=O)NC2(CC)CCN(C(=O)COC(C)C)C2)CC(c2ccccc2F)=NO1 c1(C(C)=O)cc(S(=O)(=O)NCC2(NC(=O)C(C)C)CC2)ccc1C.C1C(=O)N1 Cc1cc(Br)cc(C(N2CCC(CN(C)C(C3CC34CC4)=O)C2)=O)c1C N1(C(C(C2CN(C(c3cc(F)ccc3C)=O)C2)OC)=O)CCn2ncc(O)c2C1 c1(C(=O)NCC(c2ccccc2)N(C(C2C(C=C)C2)=O)C)cc2nc(C)sc2[nH]1 c1(C(CNC(C(C)OCC#C)=O)NC(=O)C(C)(F)F)cccc(Cl)c1Cl N1(C(CCOCCC)=O)CCC(C2CC(NC(=O)Cc3cc(C(C)C)no3)C2)C1 c1(C(N2CCC(NC(c3c(F)cccc3F)=O)C(O)C2)=O)cc2ncccc2[nH]1 CN=c1[nH]nc(CC(=O)NC2CC(CCNC(=O)CC3CCCC3C)C2)s1 c1(CC)ccc(-c2cc(C(=O)NC3(CNC(=O)C(C)C(C)O)CCC3)no2)cc1 C1(NC(c2ccc(O)cc2)=O)CCCCN(C(=O)Cc2cccc(Cl)n2)C1 c1(COC)nc(NCC2(COC)CCCCC2)cc(=NCc2nn(C)cc2Br)[nH]1 C(CC(C)(C)C)(C(=O)NCCCN(C1CCCC1)C(C1CCC(=O)N1)=O)OC C1(CNC(CC(=C)C)=O)(COC)CCCN1C(c1ccccc1C(C)=O)=O C(=O)(C(C)(C)C(C)O)NCC1(F)CC(NC(c2c(OC)cncc2)=O)C1 N1(C(C(C)C(C)n2cccn2)=O)CC2CCN(C(=O)CN(C)C)CC12 CC(C1=CCCCC1)NC(c1ccccc1)C1CCC1 N1(C(CC2CC(C(C)(C)C)C2)=O)CCN(C(=O)C=Cc2nccs2)C(CO)C1 c1(C(=O)NCC2(OC)CCN(C(CC=C=C)=O)CC2)ccc(S(N)(=O)=O)cn1 c1(OC(C(=O)NCC(n2cc(C(CC)N(C)C)nn2)C)CC)ccccc1F c1(C(N2CCC(O)(CNC(C3CC(CCO)C3)=O)C2)=O)c[nH]nc1[N+](=O)[O-] C1(=CCNC(C=C2CCN(C)C2)=O)CCN(C(=O)C(C)(C)C2CCOC2)CC1 N1(C(COCCC(C)C)=O)CC(F)CC1CNC(c1ccc(OC(C)=O)cc1)=O CC1(C)CN(C(=O)CC2CCS(=O)(=O)C2)CCC1NC(C1CC(n2cnnc2)C1)=O C1(C(=O)NCc2n(C)ccc2)CC(F)CN(C(c2ccc(I)c(O)c2)=O)C1 CC(CC(=O)NC1C2CC1N(C(c1ccc3ncnn3c1)=O)C2C)CC(C)(C)C C12(NC(C3CC4CCC3O4)=O)CCCC1N(C(c1ccoc1Br)=O)CC2 Cc1cc(F)ncc1NC(C1COCCN(C(=O)CC2(N(C)C)CCC2)C1)=O c1(OCC)cccc(C(N2CC3C(C2)N3C(c2cc(C)cc(O)c2)=O)=O)c1F N1(C(C2(F)C(C)OCC2)=O)CC=C(C(=O)N2CCN(C3CCC3)CC2)C1 c1(C(=O)NC(C)C(CO)NC(=O)CC(C)(C)C)cc(Cl)c(F)cc1[N+](=O)[O-] C1(NC(C2C(C)=CCS2)=O)CCN(C(c2ccc(O)nc2)=O)CCC1CO CCC(CC)C(C(=O)NCC(O)CN(C(=O)C(c1c(C)noc1C)(C)C)C)OC c1(OC(C)C)cncc(S(=O)(=O)NC2(CO)CCCC2)c1 n1(CC=C)nnnc1C(CCC=C(C)C)NCC1CC1(Br)Br CCC(C)CCC(=O)NC1CCCN(C(=O)COC(F)(F)F)CC1 n1(CC(C)C)ccc(CC(=O)NCC2CCC(NC(=O)CCSC(F)(F)F)C2)n1 C1(COC)(CNC(C2OCCC2NC(=O)Cc2ccc(F)nc2)=O)CC2CC2C1 C12(NC(C)=O)CCCC(CN(C(=O)CCNC(C3CCCCCC3)=O)C1)C2 c1(NC(C2CC(NC(C(c3cnn(C)c3)C)=O)C2)=O)cnc(Cl)nc1 N1(C(C2C(C#C)C2)=O)CC(C)C(C)(CNC(c2cc(OC)nc(OC)c2)=O)C1 CCC(C(=O)N(C)CCOCCC(=O)NCC1CCOC1=O)NC(C)=O C(CCCCCN(C(=O)CC1CCOC1C)C)NC(COCCCC(C)C)=O C#CCCCC(=O)NCC1C2CN(C(=O)C(O)CCC)CC12 n1(CC(=O)NC2C(NC(CCC=C)=O)CC2)c(=O)n(C)c(=O)c2ccccc12 c1(C(=O)NC(C2(C(=O)NCCOCCC=C)CCC2)C)coc(COC)n1 c1(NC(=O)NC(C(C)C)COc2ccc(F)nc2)ccc(F)cc1Cl C(CNC(c1cc(C(F)F)no1)=O)(CC(F)(F)F)NC(C1CCC(=O)C1)=O C(=O)(C1=NOC(C)(C)C1)NC(C(=O)N(c1ccccc1O)CC)CC(C)C Cc1ccc(CC(N2CCCC(NC(C3(C4CC4)CC3)=O)C2)=O)cc1Cl c1(C(N2CC(N(C(C3CCCN(C(=O)OC)C3)=O)C)C2)=O)ncc2ccccn12 CC1(CNC(c2ccncc2F)=O)CCCN(C(c2ccsc2)=O)C1 N1(C(C(n2ccc(C)n2)C)=O)CCN(C(=O)CN2CC3CC3C2)C(C2CCC2)C1 CC(CN(C)C(c1nc[nH]c1C(F)(F)F)=O)N=c1[nH]c(Cl)nc2c1SCC2 C12CCN(CC1C)C(=O)NC1C2C1(C)C.c1(C(C)C)csc(C(=O)NC2CC2)n1 c1(C(=O)OC(C2CC(NNCC(=O)N(CC)CC3CCCO3)C2)=O)occc1Br C1(CC(N2CCC(NC(C3N(CCC)CCCC3)=O)CC2)=O)CCCC(C)(C)C1 N1(C(CC(CC(C)C)O)=O)CC2N(C(=O)C(N)=O)CCC2(C)C1 Cc1cc(C(=O)NCC2CCC(F)(CNC(=O)C(C)CC3CCC3)C2)ccn1 N1(Cc2nnc(CC)s2)CCC(NC(c2csc(-c3cn[nH]c3)n2)=O)C(O)C1 N1(C(c2noc(CC)c2C)=O)CC(C)CN(c2ncc(C(C)(C)O)cn2)C(C)C1 C1(O)(CNC(C(C#C)(C)C)=O)CCCN(C(c2ccc(N)cc2C)=O)CC1 c1(CC(N2C3CC(NC(CSC)=O)C2CC3)=O)nc2ccccc2[nH]1 C(=O)(CCCCSC)N1CC(F)(CNC(C2CCN(C(CC)=O)C2)=O)C1 C=CCC(C(=O)N1CCC(NC(=O)CN(CC(C)(C)C)C)C(O)C1)C(C)C C1(N(C)C)CCCC(N=c2nc(N3CC4CCCC(C4)C3)c3ncccc3[nH]2)C1 C1(CNC(=O)CCN2CCOC2=O)CN(C(c2ncsc2Br)=O)CCO1 N1(CC2CCC(CCC)CC2)CCCC(C)(O)C1 c1(OC)ccc(Br)cc1CN1CCC1C(=O)Nc1ccc(SC)c(F)c1 C=CCC(C(=O)NC1CCN(CCNC(=O)C#CC(C)C)CC1)NC(C)=O N1(C(C(C=C)CC)=O)C(C(=O)NCC(C)Cn2ccnc2)CC2CCCC12 N1(C(C2CCN(C(C3(OC)CCC3)=O)CC2)=O)CCC(N=[N+]=[N-])C(O)C1 c1(CN(C)C)cccc(-c2cnccc2C(N2CCC(CCN)C2)=O)c1 C1(NC(CSC(CC)C)=O)CCOCC1NC(=O)CN1CCC(C)CC1 CC#CCC(C(=O)NCC(C)(C)C(C)(F)F)NC(=O)C(F)=CC1CC1 C1(C(=O)NC2CC(F)(CNC(c3c(C)cc(F)cc3)=O)C2)CN2CCCN1CC2 N1(C(C2N(C(C(CC)O)=O)CSC2)=O)CCCC1C=CC(=O)NC C1(=CC(=O)NC2C(NC(C3(OCC)CCOC3)=O)CCC2)CCCCCC1(F)F c1(NC(Cc2nnc(C)o2)=O)ccc(NC(=O)C(C)(C)C2CCC2)cc1C c1(C(=O)NC2CCN(C(C(CC)OCC)=O)C2C)cc(O)nc(C)n1 C1(NC(C(C)O)=O)C2CCC(C2)C1C(=O)NCCCC(C)(C)CO CCC(CN(C)C)C(=O)N(C1CCCC1)CCNC(=O)C(C(C)C)SC N1(C(c2nn(CC)c(C)c2)=O)CCC2CCC(NC(=O)CCc3cn(C)nn3)C12 C1(C)(C(=O)NCC2N(C(C(c3cccc(C)c3)=O)=O)CC2)CCCNC1=O c1(C(N2C(C(C)C)CN(C(=O)C(C)(C)CF)CC2)=O)cnc2[nH]ccc2n1 Cc1cc(N2CCCC3(C=CCO3)C2)nc(=NCCCC(C)(F)F)[nH]1 C1(C(=O)NC(C)CCNC(=O)CCCn2ccnc2)CC2CCC(C1)N2C1CC1 N1(C(CC(COC)C)=O)CC(NC(=O)C=Cc2ccc(O)cc2)C(C2CC2)C1 N1(C(C2C3CC=CCC23)C(=O)NCC=C)CC(C)(C)OC2(CCOC2)C1 N1(C(CCNC(C)=O)=O)CCC(C)C(NC(C2CC(O)C2)=O)C1 C1(C(N2CCC(CN(C)C)C2)=O)CN(C(c2sccc2CO)=O)CCO1 C=C(C)CC(C(=O)N1CCCCC1C(C)NC(c1nc(=O)n(C)[nH]1)=O)OC C1(C)(CCNC(CNC(CCC)=O)=O)CCN(C(=O)CCCc2ccccc2)C1 N1(C(C(C)SCC)=O)CCN(C(=O)C(CC2CCCCC2)OC)C2(CCC2)C1 S(=O)(=O)(c1cccc(C(=O)NC2C=CCCC2)c1)NC(c1c(C)cccc1)C1CC1 Cc1cccnc1NC(c1sccc1NC(c1cccc(-n2ccnc2)c1)=O)=O c1(OC)ccc(N)c(C(=O)NC2CCC(NC(=O)C(c3ccccc3)O)CC2)c1 Cc1cccc(C)c1CC(=O)NCC(C1CCOC1)NC(C1(CO)CCCC1)=O C1(C(=O)NC2CC(C#N)C2)CC(NC(C2CNC(=O)N2)=O)C12CCC2 c1(CC(=O)NC(CC)(C)C)nn(C)cc1Br.C12CN(C1)C2=O N1(C(CCCOC)=O)CCCC(O)(CNC(c2cnn(CCC(F)(F)F)c2)=O)CC1 CCCC(C)(CC)C(=O)N1CCC2(CC(NC(=O)C(F)Cc3ccccc3)C2)C1 CCC(C)C(C)(O)CNCCCOCc1ccccn1 C(C(N=[N+]=[N-])C(=O)NC(C)C=CC(=O)NCCOC1CCC1)OCC Cc1ccc(C(C)C(=O)NC2CC(CNC(=O)Cc3ccccn3)C2)cc1 N1(C(C(CC)C#N)=O)CCC2CC(NC(=O)CCOCC3CCCO3)CCC2C1 c1(C(=O)N=c2nc[nH]n2-c2ccccn2)cc2c(s1)CCNC2 c1(N(C(Cc2ccc(F)cc2F)CO)C)ccc(S(=O)(=O)NCC(Cl)Cl)c(Br)c1 C1(NC(c2cc(C)[nH]n2)=O)CC2(C1)CC2C(=O)NC(C)CC(C)C C(=O)(CCCCCC(=O)NCCN(C(=O)CCNS(C)(=O)=O)C1CC1)OCC C1(OC)C(NC(C2(NC(C3CC4CCC4C3)=O)CCN(C)C2)=O)CC12CCC2 C=C1CCN(C(c2oc(C)cc2C)=O)C(C(=O)NCc2cnc(C)n2C)C1 C1(CNC(c2c(COC)scc2)=O)C(C)CCCN1C(c1sccc1C)=O N1(C(C(C)OCC=C)=O)CC(F)CC1C(=O)Nc1cc(C(=O)OC)nn1C C1(NC(C2C3(CC(NC(c4ccc(SC)o4)=O)C3)C2)=O)CCC(=O)N(C)C1=O c1(C(=O)NCC2CN(C(C3CCC(=O)O3)=O)CC23CC3)n[nH]c2cccnc12 c1(CC)cc(OC)cc(OC)c1C(=O)NCC(C)CN(C)C(C1CCCS1)=O c1(C(N2CC(NC(C3N(C)CCOC3)=O)C(C)(C)C2)=O)cccc2c1nnn2C C=C(C)CC(C(=O)NC1(CCC)CCCN(C(=O)CC2CCCN2C)C1)OC c1(C(N2C(C(C)(C)O)CC2)=O)cc(=N)[nH]c(Cl)n1 C(C(F)(F)C(=O)NC1CCCN(C(c2ncsc2-c2ccccn2)=O)C1)N(C)C c1(NC2C(NC(C3CC3F)=O)CCC2)ccc2nc(C(F)(F)F)sc2c1 Cc1cccc(C(N2CCC2CNC(=O)Cc2cscc2Br)=O)c1C n1(CCC)ccc(C(=O)NCc2cc(C(N3CCC3CC)=O)n[nH]2)n1 C(c1cnn(C)c1)=CC(=O)N(C(C(=O)NCCOC)C)C C=CCC(C(=O)NC(CNC(=O)CCOCCOC)CC=C)C(C)C c1(C(=O)NCC2CC(NC(CNC(CC)=O)=O)C2)ccc2[nH]ccc(=O)c2c1 c1(C(N2C(CNC(c3c(C#C)cnn3C)=O)CC2)=O)ccc2nc(O)oc2c1 Cc1cnn(C)c1CC(=O)NC1C=CCN(C(=O)CC(C2CC2)C2CC2)C1 C12(CNC(CS(CC)=O)=O)CCC(CC1)CN2C(c1cn2c(n1)CCCC2)=O C1(NC(C2C(CC)CCC2)=O)CC2CCC(C1)N2C(=O)CNC(=O)C(F)(F)F N1(C(c2c(C)nn[nH]2)=O)CC(CNC(C2CCCC3(CC3)C2)=O)C2(CC2)C1 CCC(F)(F)CC(=O)NC1CC2CCC1N2C(C1(C)CCCC1)=O c1(C(N(c2cnn(C)c2)CC)=O)cccc2c1C(=O)N(c1ccc(Cl)cc1)C2=O c1(OC)cc(C(=O)NCc2ncc[nH]2)c(NCc2ccc(CC(C)C)cc2)cn1 C(=O)(NNc1c(F)cccc1I)C1CC(=O)N(C(C)C)C1(C)C c1(C(N2CCC(C)(NC(C(C3CCC3)OCC)=O)CC2)=O)ccc(S(C)(=O)=O)[nH]1 C#CCCC(N)C(=O)N1CC(CC)C(CCO)C1 N12CCC(CC1)C2.N1(C(CC)C(N)=O)CCOC(c2nnnn2C)C1 C1(C(=O)NCC#CCNC(c2coc(-c3cccnc3)n2)=O)CC=CCC1 C1(CNC(C2(CC#C)CCCC2)=O)C2CN(C(=O)CN3CCC(C)C3)CC12 N1(C(C2(C=C)CCN(C(C(C(CC)C)N(C)C)=O)C2)=O)Cc2ccc(C)cc2C1 C1(C(=O)OC(C)(C)C)CN(C(=O)C(=O)NC2CCSC2)C1 CC(C(=O)NCCN(C1CCCC1)C(=O)CSc1nncs1)=C1CCCC1 c1(N(C)CC2CCCS2)nccc(=NCCn2cnc3c2CCCC3)[nH]1 n1(CCC)nccc1C(=O)N(CCNC(C1(CF)COC1)=O)Cc1ccccc1 CC(C)C#CC(=O)N1CCCC(CNC(c2n[nH]c(C(C)(C)C)n2)=O)C1 CCC(CC)C(F)C(=O)NC(C1(O)CCCCC1)C(=O)NCC(C)C1CCC1 c1(C(=O)NC(C(=O)NC(C(=O)NC)CC2CC2)C2CC2)nnn(C)c1N Cc1nc(N2CCCCC(NC(c3sccc3Br)=O)C2)c2ccccc2n1 N1(C(Cc2cccc(CC)c2)=O)CC2CC(C1)CN(C(c1ccnnc1O)=O)C2 C(CCCCCNC(c1ccc(OCC(F)F)nc1)=O)NC(C(CC)C)=O C1(C(=O)NCc2ccc(C)nc2)CCC2(CC2)N1C(C1CCN(C)C1)=O c1(C(N(CCCNC(C(C)NS(CC)(=O)=O)=O)CCO)=O)ncc(C)cn1 C1(NC(CCOCCOC)=O)(CO)CCCN(C(=O)Cc2cn[nH]c2)C1 C1(C(N2CCOC3CC23)=O)C2CCC1CN(C(=O)CCc1cccnc1)C2 C#Cc1ccc(C(=O)NC(CO)C(C)NC(=O)CCC(C)CN(C)C)cc1 C1(C(N2CC(C(=O)NC(C=C)C3CCC3)C(CC)C2)=O)CC2(CCC2O)C1 C1(C(N2CCC(C(C)NC(=O)C=CC(=O)NC3CC3)C2)=O)NC(=O)CC1C C1(NC(CSCC=C)=O)CN(C(=O)Cn2cnc(Br)n2)C2(CCOC2)C1 c1(COC(c2cc(N)c(F)cc2Cl)=O)ccc(Cl)c2cccnc12 C1(NC(C2(CNC(C(COC)COC)=O)CC23CCC3)=O)CCc2ncnn2C1 n1(C(CC)C)nc(C(N2CCCC2(C)CNC(C2(C)CC(C)C2)=O)=O)cc1C N1(C(C=C(COC)C)=O)CCC(F)(F)C(CNC(=O)C(O)Cc2ccccn2)C1 C1(CC)CN(C(c2coc(Cl)c2)=O)CCC1NC(=O)Cc1ccc(C)o1 c1(-c2cc(NC(c3cccc(Cl)c3F)=O)sc2)ccc2nc[nH]c2c1 N1(C(C2N(C)C(=O)OC2)=O)CC2CN(C(=O)CCC3(C)CCC(=O)N3)CC2C1 CC1CCc2onc(C(=O)NCC(C3CC3)NC(c3cc(N)cnc3Cl)=O)c2C1 N1(C(=O)Cn2nnnc2C2CC2)CCC2(C1)CN(C(C1C3CCC(=O)C13)=O)C2 N1(C(C(C)CC2CC2)=O)CC2COCC(C1)C2NC(=O)C(F)Br N1(C(c2cnn(CC)n2)=O)CCCCC1C(C)NC(c1cnc(C(C)(F)F)s1)=O C12(NC(C(C)=CC)=O)CCC(CC1)N(C(=O)COCc1ccccn1)C2 C1(C(N2CC(NC(Cc3c(OC)cccc3)=O)C(C)C2)=O)CC2(C1)CC(C)(C)C2 C12(NC(C3=CCCC3C)=O)CC3CCC(C1C2)N3C(=O)CCCCC(N)=O C1(C(N2C(CNC(C=Cc3nnn(C)n3)=O)CC(F)C2)=O)CCCC(C)(C)O1 c1(C(N(CCC)CCNC(c2cc(C)ns2)=O)C)cccc([N+](=O)[O-])c1 c1(-c2cc(C(=O)NC(CNC(C(C)OCC=C)=O)(C)C)n[nH]2)ccc(O)cc1 CC1COC2(C1)CN(C(C1CCN(C(c3ocnc3C3CC3)=O)CC1)=O)C2 C1(C(=O)NC23CC(CNC(C4(CN(C)C)CC4)=O)(C2)C3)CCC2(CCC2)CO1 N1(C(CN(C)C(c2cc(Cl)c(F)cc2Cl)=O)=O)CC2CC(NC(C)(C)C)CC1C2 C(=O)(C1=CCCCC1C)NCC1(CC(=O)NCC(N(OCC)C)=O)CC1 C#CC(C)(C)C(=O)NCCN(C(=O)CC(C)CN(C)C)CCCN(C)C c1(OC)ccc(NC(C2CC(F)CN2C(c2cnc(N(C)C)o2)=O)=O)cc1 C1(C(=O)NC(C)(CNC(=O)CCc2ccncn2)C2CC2)CC(O)CN1C(N)=O C1(C(NOCCC)=O)CCOCC1NC(c1cn(C)nc1CC)=O c1(NC(C2C3CN(Cc4ccc(OC)nn4)C2C3)=O)ccnc(Cl)c1I N1(CC)CCN(C(=O)Nc2ccc(-c3ccccc3)cc2)CC1CC#N C1(C(N(C)CCNC(c2csc(-c3cccs3)n2)=O)=O)CCc2c(ncn2C)C1 c1(C(N2C(C(C)C)CN(Cc3ccccn3)CC2)=O)cn2ccccc2n1 C1(C(N(C(CN(CCCCCC)C)=O)CCOC)=O)CCC=CCCC1 CCCN=C(NCC1CC(O)CCO1)N1CCC(CC)(Cc2ccccc2)CC1 c1(N2CCC(C)OC(C)C2)ncnc2c1ncn2CCN1CCCCCC1 c1(CC(N2CCCCC(NC(c3c(C)cnnc3)=O)C2)=O)nc(F)c(F)cc1F N1(Cc2scc(C)n2)CC(F)CC1C(=O)NCc1ccc(F)nc1 CN1CC(NC(=O)C=CCNC(C2(F)CC=CCC2)=O)C(=O)N1 C1(C(=O)Nc2c(OCC)ccnc2)CC(C)CN(C(c2ccccc2Cl)=O)C1 C1(CNC(c2cc(C)n(C)n2)=O)CC2CCC1N(C(=O)C(C)CS(C)(=O)=O)C2 C1(CC=C)(C(=O)N(CC(=O)NC)C)CCN(C(=O)CC2CCCOC2)CC1 C(=O)(C1Cc2ccc(Cl)cc21)N1CCN(C(C2CCCCC2(F)F)=O)CC1CO C1(F)(C(N(CC(C)N(C)C(c2sccc2C#N)=O)C)=O)CCCN(C)C1 C1(n2cc(CN3C(C(=O)O)CCCC3)nn2)C2CCC1C(OC(F)(F)F)C2 c1(OC)ccc(Cl)c(F)c1C(=O)NCCCNC(=O)CSCc1cscn1 N1(C(CC(C(C)C)(F)F)=O)CCC2(CCCN2C(=O)CS(C)(=O)=O)CC1 C(=O)(C1CCCc2ncnn21)NC(C)(C)CCNC(C1CC2C=CC1C2)=O N1(C(C(CCC)C)=O)CCC(O)(CN(C)C(c2cc(Br)cn2CC)=O)CC1 c1(C(=O)NCC2CCC(NC(C3CCC(C)CC3)=O)C2)cc2[nH]ccc2s1 Cc1ccc(C)c(C(N2CCC(CN(C)C(C3(C)CC=CCC3)=O)C2)=O)c1O CC(C)C(O)C(=O)N1CCC(C)(CNC(=O)CN2CCCC2)C1 C1(N(C(c2cn(CC)nn2)=O)C)CN(C(c2ccncc2C)=O)CC12CC2 CC(C)(F)C(C)(C)N(C(c1cccc(CC2CCNCC2)n1)=O)Cc1cccnc1 C1(C(C)C)CCN(C(c2cnc(N(C)C)cn2)=O)C(CNC(=O)CCCSC)C1 c1(-c2cn(CCC3CN(C(=O)Cn4cnnc4)C3)nn2)cccc2c1OCC2 N1(C(C(C)(C)C2CCC2)=O)CCN(C(=O)Cc2cocn2)C2CCCCC2C1 c1(COC)cccnc1C(=O)N(C1CCN(C(=O)C(C)C2CCC2)C1)C C(CC[Si](C)(C)C)n1c(C2(NC(C(=O)OC)CSC)CCSC2)nnn1 N1(C(CC(COC)C)=O)CCC(NC(c2cnc(O)c(OC)c2)=O)CC(C)(C)C1 C(CCOC)(C(=O)NCC1CNC(=O)C1)NC(c1cc(CC)sn1)=O Cc1ccc([N+](=O)[O-])cc1C(=O)NC1CCN(C(c2cnc(N)cn2)=O)CC1O c1(OCC)cc(C(=O)NC2CC2C(=O)NCCC2CCCC2)ccn1 CN1CC2(CC(NC(C3CC(NC(c4cc5n(n4)CCC5)=O)C3)=O)C2)C1 CC1=C(C(=O)NCC2CC(NC(=O)C=CC(=O)N(C)C)C2(C)C)COCC1 c1(OC)cc(C)c(CNc2cccnc2C(=O)NC(C)C(N)=O)c(C)c1 c1(C(=O)NC2(CCNC(c3c(CC)cc(F)cc3)=O)CC2)cc2c(ccn2C)[nH]1 Cc1nn(C)c(F)c1C(=O)NCCC1CN(C(=O)C(F)Cc2ccccc2)C1 Cc1cc(Cl)c(C(N2CCC(NC(=O)CCN3C(=O)CCC3=O)C2C)=O)cn1 C(=O)(CCC(CF)CF)NC(CC)(C)CNC(=O)C=C1CCOCC1 CCCC(C(O)C(=O)NC(c1n[nH]c(C)n1)(C)C)NC(C1CCC2(CC2)C1)=O C1(C(=O)NCc2cc(C)c(O)cc2)CCCN1NC(=O)C(C)C1CCOCC1 N1(C(COCC)=O)CC(C)CN(C(=O)Cc2ccc([N+](=O)[O-])cc2F)C(C)C1 N#Cc1c(F)cc(CN2CCCC2CC(=O)NCCC(=O)NC(C)(C)C)cc1F Cc1cc(CCC(=O)NCC2CC(NC(=O)C(F)=C3CCCC3)C2)c(C)s1 CC(C)(C(=O)N(CCCCN(C(=O)CCCc1ccc(N)cc1)C)C)C(F)(F)F C1(CC(=O)NCCN(C(CC)C)C)CCCN1C(C1CCC(N(C)C)C1)=O c1(C(N2CC3(CC3)CC2C)C(=O)NC(C(=O)OC)C)ccc2ncsc2c1 C1(C(N(C(CC)CC)CCO)=O)COC2(C1)CN(C(C1CCC(F)(F)C1)=O)C2 Cc1ncnc(C)c1C(=O)NC1CCC(CNC(=O)C(F)F)C1 c1(CC(=O)NCC2OCCN(C(c3c(OCC)ccs3)=O)C2)cc(O)nc(O)n1 C#CC1(NS(=O)(=O)CC2CCC(C)N(C(=O)OC(C)(C)C)C2)CCCCC1 C(CCC(C)(C)C(=O)NC1CN(C(=O)OC)CC1SC)NC(CC1C(CC)C1)=O C1(C(N2CCN(c3ccccc3Cl)CC2)C(=O)NCC=C)CC2(CCCO2)C1 c1(C(N2CC(NC(c3ccc(O)nc3)=O)CC(OC)C2)=O)csc(S(C)(=O)=O)c1 N1(C(c2c(C=C)cnn2C)=O)CCC2(C1)CN(C(=O)CCC(=C)C)CCO2 CCC(CC(=O)NC1CC1NC(C1(C#N)CCCC1)=O)CC(F)(F)F C1(F)(CN(C)C)CCCN(C(=O)C(C)(C)CNC(C2CCC(=O)N2)=O)C1 C1(CC(=O)OC)CCCCN1C(=O)CC(C)n1ccnc1N Cc1cc(N2CC(CO)C(C3CC3)C2)n2nc(C(F)(F)F)nc2n1 C12(C(N3CC(C)C(NC(=O)C=CC4COC(C)(C)O4)C3)=O)CCCC1CCC2 C1(CC(=O)N(CC(C)C)CCO)CCCN(C(C2OCCC2(C)C)=O)CC1 C1(CC)CN(C(c2nocc2C(C)(C)C)=O)CCC1NC(=O)C=C(C)C c1(C(=O)NCC2CC(F)CN2C(c2cc(CO)on2)=O)cc2c(s1)CCOC2 n1(CC(N2CC(CC(C)NC(c3cccnc3CO)=O)C2)=O)ccccc1=O c1(NC(c2n[nH]c3ccc(I)cc23)=O)c(C(=O)O)oc2ccccc12 N1(C(C=C(CC)CC)=O)CCCC2(CCCN2C(C2CCCC3(CC3)C2)=O)C1 c1(C(=O)NCC2(CO)CC2)cc2c3c(ccc2[nH]1)N(C(=O)CCC1CC1)CC3 c1(CC)oc(C)cc1C(=O)N(CCC(C)NC(C1CCC(C(N)=O)C1)=O)C CCC(C(=O)NC1CCCCC1NC(c1cnn(C(C)(C)C)c1Cl)=O)C(C)C c1(CNC(C2CCN(C(c3cc(C)no3)=O)C2)=O)ccc([N+](=O)[O-])cc1C c1(NCC2CCCN(C(CCC(=O)N(C)C)=O)C2)nc2ccccc2o1 C12(C(=O)NC3CCC(CCC(N4C(C)CC4CO)=O)C3)CCC(CC1)CO2 c1(CC(C)C)ccc(C(C)C(=O)N(C(c2ccco2)C)Cc2ccccn2)cc1 CCC(C)C(=O)N1CC(NC(C2CC(F)(F)C2)=O)C1 N1(C(Cn2cc(CC(=O)Nc3ccc(C)cc3)nn2)=O)CCC(C)(C)C1C C(=O)(CCCC(C)CC)NCC1(NC(C2C(C=C)C2)=O)CC(C(F)(F)F)(OC)C1 N1(C(CN=S(C)(C)=O)=O)CCC2(CCCN2C(C2CC(O)C2)=O)CC1 c1(C(N2CCC(N(C(C=CC=CCC)=O)CC)C2)=O)ccc(F)c(C(=O)NC)c1 c1(C(=O)NCCCCNC(C(CCC)O)=O)ccc2c(c1)NC(=O)CN2C c1(C(N(C2CCN(C(C3C(CC)C3)=O)C2)C)=O)cncc(N2CCOCC2)c1 c1(OC)ncnc2cc(-c3nc4c(s3)CCN(C(C3(C(C)C)CC3)=O)C4)ccc12 c1(C(=O)NCC(C)N(C(=O)CCC2CC2)CC)cc(C(C)C)n(C)c1C N1(C(C2C(C)(C)C2(C)C)=O)CC2(CC(NC(c3cc4c(s3)CCSC4)=O)CO2)C1 c1(C(=O)NC(C)CN(C(=O)C(O)C2CCCC2)C)cnc(-c2ccoc2)s1 c1(COC)cc(=NCC(C)(C(C)C)NC(c2cc(O)n(C)n2)=O)[nH]c(C(C)C)n1 Cc1cc(C(N2CCC3(CC3C(=O)NCC(=O)OCC3CC3)C2)=O)c(C)cn1 C(CCC(=O)NC(CO)C(C)NC(=O)CCN(C1CC1)C(C)C)=CC(C)C CC1(C)CN(CC(=O)NCC2CC2C(N2CC(c3ccon3)C2)=O)C1 c1(CC)cccc(C(N2CCOCC2CNC(c2cc(C)c(Br)s2)=O)=O)n1 O=C1CC(C2CC2)(C(N2CCC(CNC(C3CC4CCC3CC4)=O)C(O)C2)=O)C1 C1(NC(c2cnc(C(C)OC)s2)=O)C2CCC1N(C(=O)C(C)(CC)CC)C2 C(=O)(C(C)CC(F)F)N(C1CCN(C(=O)CC(C)(C)C#N)C1)CCC C1(C(=O)NCCN(C(=O)CCC2CCCC(O)C2)C)(N(C)C)CCCCC1 C1(NC(C2(CN(C)C)CC2)=O)CC2CC(NC(=O)CCc3cc(Cl)cs3)CC2C1 c1(C(N2C3CCC2CN(C)C3)C(=O)NCC)ccc(Cl)c(Cl)c1Cl c1(C(=O)NC2(COC)CN(C(=O)CC(C)(C)OC)C2)cc[nH]c2nccc1-2 N1(C(Cc2nc(C)c(C)[nH]2)=O)CCCC(C)C1CNC(=O)CCC1CCC(=O)C1 C1(NC(C(C2CCC2)OC)=O)CCCC1NC(=O)C(c1cccnc1)OC c1(SCC)ccc([N+](=O)[O-])cc1C(=O)NC(C)CN(C)C(c1nnc(C)s1)=O c1(C(=O)NCCC2(NC(C=CSC)=O)CCCC2)cc([N+](=O)[O-])c(C)cc1C N1(c2c(C)cccc2[N+](=O)[O-])CC2C3CCC(C2C1)N(C(C1CC(F)(F)C1)=O)C3 c1(NC(c2cc(Br)ccc2-c2nnnn2C2CC2)=O)c(Br)ccc2ncccc12 c1(C(=O)NC(C(=O)NC(C)C(C)C)Cn2cccn2)cc(O)ncc1F C1(C(NOCC(=O)NCCN(C(C)C)C(C)C)=O)CC2CCCC2C1 c1(C(N2CC(C)(C(=O)Nc3c(O)ccc(CC)c3)C2)=O)cccc2c1CCCC2 c1(C(=O)NCCCCN(C)C(C2CCCC(=O)N2)=O)cccc2c1CCO2 O=C(Cc1ccccc1I)N=c1cc(Cl)nc(Cl)[nH]1 CC(C)CC(C)(O)C(=O)N1CCC2(CC1)CC2NC(=O)COC(F)F CC1(C)CCC(Cl)=C(C(=O)NC(c2cccnc2)CCc2ccccc2)C1 c1(C(CC(C)C)C)noc(C2c3c[nH]nc3CCC2C)n1 Cc1cc(CC(=O)NC(CNC(C2CCCS2(=O)=O)=O)CO)cc(Br)c1 CCCCC(F)C(=O)NC1CCOC(C(N2CCC2CF)=O)C1 N1(C(Cc2c(C(=O)OC)cccc2)=O)CCN(C(C2CC2C)=O)CC1C C12(CCCC1C)c1ccn(n1)C1CN(C1)C(=O)N2.C1COCCO1.CC.OC c1(NC(C=C)C)nc(N2CC(C#N)C3(CCC3)C2)nc2c1ncn2C N1(C(c2ncn(CC)c2)=O)CCCC(N(C)C(c2cc(C3CCC3)nn2C)=O)C1 C1(CC(N2CCCC(C(=O)OC)C2C)=O)CCc2ccccc2C1=O Cc1cccc2[nH]cc(CNc3ccc(C(C)C)cc3)c12 n1(C(CC)(C)C)nnnc1C(c1cnnn1CC)NCC1CC1 N1(C(c2c(N)cncc2)=O)CC2(CCC2NC(=O)Cc2cnns2)C1 c1(OC)cc(NC(c2n[nH]cc2NCc2ccccc2Br)=O)cnc1Cl Cc1ccc(CC(=O)NCC(C)(C)NC(=O)C(F)C2CC2)cn1 N1(C(CC=C)=O)CCc2c(C(=O)N(CC(O)CO)C(C)C)cccc2C1 C(=O)(CCCCC(C)(C)C)NC(CN(C(=O)C(O)C(F)(F)F)CC)C CCCC(C)CCCC(=O)NC1COCCN(C(=O)C=CC(=O)OC(C)(C)C)C1 C1(C(N2CCCC(CCC#C)C2)=O)C(C2CC2)CCN1C(c1csc(O)n1)=O C1(C(=O)NCCN(CCOC)C)CN(C(=O)C(C)n2cnnn2)CC(C)O1 CC1(C)C2CCC(C(N3CCC3CNC(C3CCCCCC3(F)F)=O)=O)C1C2 C1(C(N2CC(CN(C)C(C3CSC3)=O)C3(C2)CC3)=O)CCOCC12CCC2 O=C(C(O)C(F)F)NCC1CC(NC(c2ccccc2SC(F)(F)F)=O)C1 N1(C(C2(C)CCOCC2)=O)CCCC(NC(=O)COCC2CCCC2)C(F)C1 N1(C(COCCOCC)=O)CCC(C2(NC(c3ncc(Cl)cc3Cl)=O)CC2)CC1 c1(C(N2C(C)CC3(CC3)C2)C(=O)NCC2CCCCC2)cc2ccncc2o1 N1(C(CC(=O)NCC#C)=O)C2CCCC1CC(NC(=O)C(F)(F)CC1CC1)C2 c1(NC(CC)=O)cccc(C(=O)NC(C)CN(C)C(c2ccncc2C)=O)c1C c1(C(N(CCC#N)C2CC2)=O)scnc1C1=CCC(N2CCOCC2)CC1 N1(C(Cc2cccc(C)n2)=O)CCCC2C1CCN2C(c1ccc(Cl)c(Br)c1)=O N1(C(C(C)c2ccsc2)=O)CCC(CNC(=O)Cc2cocn2)C(F)(F)C1 N(C1=Nc2ccccc2CC1CO)Cc1cc(=N)[nH]c(Cl)n1 Cc1cc(C(N2CC3CN(C(C4CCC(=O)N4C)=O)CC3C2)=O)cc(C#N)c1 CC(C)(C)C(C)(C)C(=O)NC1CCCC1CNC(=O)COc1ccc(F)nc1 c1(C(N(C(C(C(C)C)=O)=O)C(C)(C)C(=O)OC)=O)cc2ncnc(O)c2cc1Cl c1(C(N2C(C)(C)C(C(=O)NCC3(O)CCOCC3)CC2)=O)cc2ccncc2[nH]1 Cc1cc(=NCc2cc(Br)cn2C)[nH]c(NC2CCC(CC(C)C)C2)n1 c1(CC(C(=O)NCC2N(C(c3scc(COC)c3)=O)CC2)OC)ccc(F)cc1 c1(C(=O)NCCC(C)N(C)C(c2cnn3c2OCC3)=O)cc2n(c1)CCCC2 CCC(C)C(CC(=O)N1CCCC(C)C1)NC(=O)C(O)CCC(C)C N1(C(C2(CCC)CC2)=O)CCC2CCN(c3ncnc4cccnc34)CC2C1 c1(C(N2CC(C)(C(=O)Nc3cccc(CO)n3)C2)=O)cc2n(n1)CCC2 C(CC(C)(C)C)(C(=O)N(C1CC(NC(c2cnc(Cl)c(N)c2)=O)C1)C)OC C1(OCC(N2C(CC)CCC2)=O)CCCN(C(=O)Nc2ccco2)CC1 N1(C(c2c(CNC(CCSCC)=O)ccs2)=O)CCC(F)(CO)C1 N1(C(c2c(C)nncc2)=O)CCC2CCN(c3cc(O)nc(O)n3)CC2C1 c1(OC)ccc(O)c(C(N2C(C)C3CC2C3NC(=O)Cc2ccc(O)nc2)=O)c1 N1(C(C2CC(F)CCN2C(=O)CSC2CC2)=O)CCCC(c2ccncc2)CC1 C(CO)(CCCO)NC(C1C(NC(CC2(COC)CC2)=O)COC1)=O Cc1nc(O)nc(C)c1CC(N1CCC(=CCNC(C2CSCCS2)=O)CC1)=O C1(O)(CN(C)C(c2ccoc2Br)=O)CCN(C(c2ccccc2CO)=O)C1 CN1C(=O)CSC1=CC(=O)N1CC2(C1)CN(C(c1cc(C3CC3)[nH]n1)=O)C2 C1(NC(c2n(C)ccc2)=O)CC2CN(C(C3CCC(C)(F)CC3)=O)CC12 c1(-c2cc(C(=O)NC3(CNC(CN(C)CC)=O)CCOC3)on2)ccccc1Cl C(=O)(CCC(=O)NN(C)C)N(CCOC)CCNC(=O)Cc1ccccc1C C1(C(=O)OCC)CCN(C(C2CCCN2C(=O)NC)=O)C1CC(=O)NC(C)(C)C n1(CC)cc(C2OCCC2n2cc(C3NCC3(C)C)nn2)cn1 c1(N2CCCC(OC)CC2)nc(=NCc2ccc(N)cc2C)[nH]c2ccccc12 C(=O)(CCC(C)(C)N(C)C)N1C(C(C)NC(=O)CC(O)CN(C)C)CCC1 C1(C(=O)NCC(C23CCC(CC2)C3)NC(C=CCOC)=O)CCN(C)C1=O c1ccc(Cl)cc1Cl.C(CC(=O)NCC(C)(C)NC(=O)COCCO)SCC c1(C(N2CC(CCNC(C3CC(SC)C3)=O)C2)=O)ccc2c(c1)NC(=O)C(C)O2 N1(C(C(CCC)NC(N)=O)=O)CCCC(CO)(NC(c2cc3c(s2)CCC3)=O)C1 c1(C(=O)NCC(C2(O)CCN(C(c3ccc(O)nc3)=O)C2)C)cc(Cl)ccn1 C1(SCC)C(C(N2CC(OC(C)=O)C2)=O)CCN1C(=O)CC1C(C)(C)C1(C)C C(=O)(C1=NOC2(CCC2)C1)N1CCC(C(=O)NCC2ON=C(C)C2)CC1 N1(C(C(CCOC)OC)=O)CCC(C(=O)NCC2CCCS2)CC1(C)C C(=O)(CC(C)CCC(=O)N1CCC(CNC(C2C=CC=CC=C2)=O)C12CC2)OC CC1(C)CN(C(=O)CCc2ccccc2O)CCN(C(=O)CC2C=CCC2)C1 c1(N2CCN(C(CN(C(=O)OCC)C)=O)CC2)snc(C)c1C#N C(CC1=CCN(C(C2CC(C)(C(C)(C)C)C2)=O)CC1)NC(C(C)OCCC#C)=O c1(C(N2CCCC2c2ccncn2)C(=O)NCC=C)ccc2c(c1Cl)OCO2 c1(C(=O)NCC2(C)CCCN2C(c2cnc(F)c(F)c2)=O)ccnc(Cl)c1Cl Cc1cn(CC(=O)NC2(C)CC(NC(=O)COCC3CCC3)C2)nc1C(F)(F)F c1(OC)c(C)cc(C(=O)NCC2CN(C(=O)C3=CCSC3)C3CC23)cc1C CC1(C)CC1(C)NC(=O)C(CC1CCCC1)NC(=O)C(F)CC1CCOC1 c1(C(N2C3C(NC(C4CCCCC4(F)F)=O)C(C3)C2)=O)ccc2c(c1)OCCO2 N1(C(C(C)C2CCCC2)=O)CC(C)(CCC(=O)NCCC(O)C2CCC2)C1 O=C(CS(=O)(=O)CC1CCCO1)NC1CCC(CCNC(=O)C(F)=CCCF)C1 Cc1cc(C)n(C(C)CNC(=O)Nc2cc(CSc3ccccc3)ccn2)n1 c1(OC)cnc(C(N2CC3C(CN(C(=O)CN(C4CC4)CC)C)C3C2)=O)nc1 CCCCC(C(=O)N1CCSC(CC)C1)NC(c1cn(C2CC2)cn1)=O C1(CC(=O)NCC(CN(C(c2cc(CC)no2)=O)C)O)CCCC12CC2 N1(CC2(NC(=O)OC(C)(C)C)CC(C(=O)O)C2)CCC2(COCC(CCO)O2)C1 Cc1ncccc1-n1nc(CCn2cncn2)nc1-c1ccccc1C1(C)CC1 C1(O)(CNC(=O)CC2CCCCO2)CCCN(Cc2ccc(O)c(O)c2)C1 N1(C(CCCOC)=O)CCCCC(C(=O)NC2COCC(C)(C)C2)C1 CC1(C)CCN(C(=O)C(F)C(F)(F)F)CC1CNC(C1(C(F)F)CCCC1)=O Cc1cc(C(N2CCC(NC(C3CCN(C)C3)=O)C(F)C2)=O)cnc1C c1(C(=O)NC(C2CCN(C(CCCc3onc(C)n3)=O)C2)C)ncc(F)cc1N Cc1coc(C(=O)N(C2CCN(C(c3cc(F)n(C)n3)=O)C2)CCO)c1C c1(C(N2CCC(N(C(=O)C(CC)=CC)CC#C)CC2)=O)ccc(C)nc1C O=C(C1CCc2cccc(=O)n21)NC1CN(C(=O)CCc2cc(Cl)cc(Cl)c2)C1 Cc1nc(C(=O)NC(C)CCO)sc1-c1cccnc1OC(F)F C1(C(C(=O)N(CCCc2ccco2)C)NC(C2CC2(F)Cl)=O)CC=CCC1 C12(C(=O)NC(CC)C)CCN(C(C)=O)CC1C2.c12ccc(cc1)oc2=O Cc1cc(C(N2CCCC2(C)C(=O)O)=O)n(Cc2cccc(F)c2)n1 C1(CCNC(c2c(C)snn2)=O)C(C)CCCN1C(=O)Cn1ccnc1C c1(C(C)C(=O)NCC(C)(C)NC(=O)CCP(C)(C)=O)ccc(S(N)(=O)=O)cc1 C1(C(=O)NCC2(O)CCN(C(C#CC(C)(C)O)=O)CC2)CCCCC1C1CC1 CC1CCN(C(c2ccnc(F)c2)=O)CC1NC(=O)CO Cc1c(C(=O)NCC(C)C(=O)N(C)CC2CCCCC2)cccc1C#N CS(=O)(=O)C1(C(N2CC(NC(=O)C=Cc3cscn3)C2)=O)COC(=O)C1 N1(C(c2cn(C(F)F)cn2)=O)CCC2(CCCN2C(c2ccc(Cl)nc2)=O)C1 Cc1[nH]nc(Cl)c1C(=O)NCCC(C(C)C)NC(C1CC2C=CC1C2)=O c1(C(c2nnnn2CC)NC(C(=O)NCCC)C)c(C)cc(Br)cc1F C1(Cc2nnc(N3CC(C)C(CO)CC3)n2C)COc2ccccc2O1 C(=O)(C(F)CCC(C)C)N(C(CNC(c1c(C)c(C2CC2)[nH]n1)=O)C)C N1(C(c2ccccn2)=O)CCCCC1Cn1cc(CCC2CCOC2)nn1 c1(CCNC(c2cc(F)cc(Cl)c2)=O)nc2ccccc2[nH]1 C#CCC(C)C(=O)NCCN(C(=O)COCCC(C)C)Cc1cccc(F)c1 N1(C(C(c2cccc(F)c2)C)=O)CC2(C)CN(C(C3CCC(C)O3)=O)CC2(C)C1 c1(N2CCCC(C)(NC(C(CC)c3ccccc3)=O)C2)ncc(C)cc1[N+](=O)[O-] Cc1ccc(C(=O)NC2(C3CN(C(=O)CCCc4cnccn4)C3)CC2)cc1O N1(C(c2ncc(C)[n+]([O-])c2)=O)CC2(C=C(C(=O)NC3CCCC(O)C3)CO2)C1 c1(C(=O)NC2(CNC(CC3(C)CCS(=O)(=O)N3)=O)CCC2)cnn2c1NCCC2 C1(c2c(F)ccc(F)c2)CCN(N2CCC2c2nccs2)CC1 C12(C(=O)Nc3cccc(NC(=O)CCc4nc(O)n[nH]4)c3)CCC(CF)(C1)OC2 C12(NC(c3n(C)ccc3)=O)COCCC1CN(C(c1coc(C(N)=O)c1)=O)C2 C1(C(Cn2cc(-c3n(C(C)C)ccn3)nn2)F)CCN(C(=O)C(C)(Cl)Cl)CC1 CCCCC#CC(C)(C)NC(=O)C(c1ccco1)NC(C1CC(=O)N(CC)C1)=O C(c1ccncn1)=CC(=O)NC(c1cn(C)nc1)C(=O)NCCC1CC(O)C1 n1(CC(=O)NCC2(NC(=O)COC(F)(F)F)CCC2)nc(C(F)F)cc1C(F)F N1(C(CC)=O)CCC2(CCOC2)C(CNC(c2cn(C(C)(C)C)nc2C)=O)C1 C12(C(=O)NC(C3CCN(C(=O)C=C4CCCC4)C3)(C)C)CCC(CC1)C2 c1(C(=O)NCCC(C)(C)NC(C=CCC)=O)ccc([N+](=O)[O-])cc1 C#CC(CNC(C1CN(C(C2(C3CC3)CC2)=O)CC1C)=O)C(C)C C12(CC(=O)NCC(=C)Cl)CCC1CN(C(C1CC3(C1)CC(O)C3)=O)C2 CC1(NC(c2cnnc(O)c2)=O)CCCCC1C(=O)NCCC1CC1 CCC(C)(C#N)C(=O)N1CC(O)(C(C)NC(c2ccc(C)c(Br)c2)=O)C1 N1(CCC)C(=O)CCC1C(N1CC2CC1(CNC(c1cnc(C(C)C)[nH]1)=O)C2)=O N1(C(CC2CC(SC)C2)=O)CC(C)(C)CCC1CNC(C1(C)CC(F)(F)C1)=O c1(C(N2C(CCCNC(=O)C=C3CCC3)CCCC2)=O)cccc2nc(Cl)cn12 CCCCCCCC(=O)NC1CCC12CN(C(=O)C(=Cc1c[nH]cn1)F)C2 N1(C(C2(CCCC)CC2)=O)CCCCC(NC(=O)C=Cc2ncc[nH]2)C1 S(=O)(=O)(c1cc(F)c(Br)c(F)c1)N1CC(C(=O)Nc2cn(COC)nc2)NCC1 C(c1ccnn1C)=CC(=O)NCC=CCC(=O)NC(c1cnn(C)c1)C N1(C(C)=O)CCCC(O)(CC(=O)NC2CC(F)(CNC(c3nsnc3O)=O)C2)C1 C(C1=NOC2(CCC2)C1)NC(C1N(C(c2ccc(C#C)cc2)=O)CCN(C)C1)=O c1(C(=O)NC(CC=C)CNC(=O)Cc2ccccn2)cccc(-n2cccn2)c1 c1(C(=O)NC2CN(C(C3(CC=C)COC3)=O)CC2O)cc2c(C)cc(F)cc2[nH]1 CC1COCC(CSc2nnc(C3CC3)n2-c2ccccc2Cl)O1 c1(CC(=O)NC(CNC(C2(COC)CCC(=O)N2)=O)CO)c(F)cc(F)cc1F Cc1ncc(C(N2CCC(C(C)NC(c3csc(Cl)c3Cl)=O)C2)=O)c(C2CC2)n1 c1(C(=O)N(CCn2ccnc2)Cc2ccccn2)ncoc1C1CCC1 CC(C(=O)N1CCC1CC(=O)NCC12CCCN1CCC2)S(C)(=O)=O CCCC(CCCNC(c1cncn1C)=O)NC(=O)CC1CCN(C(C)C)CC1 N1(CC(=O)NCC(CN(C(c2ccccc2)=O)CC)(C)C)CCS(=O)(=O)CC1 N1(C(C(C=C)c2ccccc2)=O)C(C)CN(C(C23CCCC2C3)=O)CC1C C=CCC(CC(=O)N1CC(N(C)C2CC2)C1)NC(=O)CC1(O)CCCC1 n1(CC(C)NC(=O)CN2CC3CC3C2)cc(C(C)(C)N(C)C)nn1 C1(CCNC(C=CC=CCC)=O)CCN(C(=O)CSCc2nccn2C)C(C)C1 c1(C(NNC(Cc2nn(C)c(O)c2)=O)=O)nc2c(s1)CCCC2 Cc1nc(N2CCC(F)(CNC(=O)CC(O)CN(C)C)CC2)cc2nncn12 N1(C(c2c(OCC)ccs2)=O)CC2CCN(c3ccncn3)CC2C1 C1(CNC(C2C(C#C)C2)=O)C2CN(C(=O)CCNc3ccccc3C(N)=O)CC12 c1(C(N(C(CN(C(COCCOCC#C)=O)C)C)C)=O)cccc(O)c1Cl CC(C1CCCCC1)=CC(=O)NC1CC(C)(CNC(=O)C2=CCSC2)C1 C(=O)(C(CNC(c1cc(Cl)ccc1C)=O)C(C)(C)C)N(CCOC)C N1(C(c2ccn(CCCC)n2)=O)CCN(C(=O)Cc2cncc(C)c2)CC12CC2 C1(N)CCCCC1N1CCCC1=O.CC1CN(C)C(=O)C2(CC2)C(=O)N1.C1(C)CC1 c1(C(N(C2CCCN(CCC)CC2)C)=O)cc(Br)cn2ncnc12 C(=O)(CC1=CCN(C)CC1)NC1C(NC(c2cc(C)no2)=O)CS(=O)(=O)C1 CC1CCCC(C(=O)NC2CCN(C(=O)CCCn3c(O)nnc3O)C(C)C2)CC1 c1(C(N2C(C(C)NC(C=CC=CCC)=O)CCCC2)=O)cc2sc(Cl)cc2[nH]1 c1(C(N2CC(CC)C(NC(c3ccc(F)cc3)=O)C2)=O)ccc2c(c1)CC(C)O2 C1(C(=O)NCC(C2CCCC2)NC(=O)Cc2c[nH]cc2CO)(CO)CC(F)(F)C1 C=CCCN=C(NCCN(S(C)(=O)=O)C)N1CCCC(C2(C)OCCO2)C1 Cc1scc(C(=O)NCC2CCCC2NC(=O)C(C(C)C)NS(C)(=O)=O)c1N C1(NC(c2n(C)nnc2)=O)CC(NC(c2nc(Cl)ccc2N)=O)C12CCC2 N1(C(c2c(C(C)(C)C)[nH]cn2)=O)CCCC(CNC(c2ccncc2Cl)=O)CC1 C1(=CC(N2C(CNC(Cc3c(C)con3)=O)CC3CC32)=O)CCC(C)(C)CC1 C1(NC(CC2(C)CC(F)(F)C2)=O)CN(C(C2CCOC(=O)CC2)=O)C2CCCC12 c1(C2CN(C(=O)NCC3CCC4(CCOCC4)O3)C2)ncc(S(=O)(=O)C(F)(F)F)cn1 C1(O)(CN(C(C2C(CCOC)C2)=O)C)CCN(C(C2(C3CC3)CCC2)=O)C1 O=C(C1=CCOCC1)NCC1CN(C(C2CCC(C(F)(F)F)O2)=O)CC1(F)F C(=O)(C(C)(C)c1cn(CCN(C)C(c2scnc2C(F)F)=O)nn1)OC c1(C(C(=O)NC)N(C2CC2)Cc2ccsc2)ccc(C(C)(C)C)o1 C1(NC(c2ccc(OCCC)cc2)=O)CCN(C(C2(CC)CCCC2)=O)CC1O N1(C(CC(CC)OC)=O)CCC(CC(=O)N(C)Cc2scnc2C)C1(C)C c1(C(N(C2CN(C(c3ccnc(Br)c3F)=O)C2)C)=O)cnc2snnc2c1 c1(C(=O)OC)cc(C(N2CCOC(CCNC(=O)C3=CCC3)C2)=O)c(C)o1 c1(OCC)ccc(C(=O)NC2CC(C)CN(C(=O)CC3(C)CCCO3)C2)cc1C C1(C(=O)NC2CCCC(CNC(c3ccnn3C)=O)C2)(OC)CS(=O)(=O)C1 c1(C(N2CCCC(CCC)(NC(=O)CN(C)C3CC3)C2)=O)ccc2ccoc2c1 N1(C(C(COC)OC)=O)CC(C)N(C(=O)CCn2nc(C)nc2C)CC1C c1(NCC2(C)N=C(C)SC2)cc(N2CCN(S(=O)(=O)CC(C)C)CC2)nc(C)n1 c1(CC(=O)NCC(CC=C)NC(=O)Cc2cc[nH]n2)ccc2oc(C)nc2c1 Cc1c(C(N2CCC(CO)C(NC(c3ccccc3Cl)=O)C2)=O)cncc1F N1(C(COc2ncc(C)s2)=O)CC2CC(NC(c3cnnc(O)c3)=O)CC1C2 C1(N2CCCC2)CCN(C)CC1.Cc1noc(C(C(C)C)N)n1 C(=O)(C1=CCCN(C(C2CCCOC2)=O)C1)NCc1cnc(C(C)C)[nH]1 c1(C(N2C(C)CC(NC(c3cn(C)nn3)=O)CC2)=O)cncc2ccccc12 C1(C)(C(=O)NCC2(COC)CCCC2)CCC(=O)NC1 C1(C(=O)OC)CCC(C(=O)NC(C)CCNC(=O)C(C)(C2CC2)OC)CC1 C(CCOC)(C(=O)NCc1ncc(CO)o1)NC(C(C)SCC)=O n1(CCC(=O)N(C)CCOC(F)F)cc(C#N)c(O)nc1=O C1(C(=O)NCC2C(NC(CSCc3ccc(C)cc3)=O)C2)OC2CCC1CC2 N1(C(CCOCC(C)(C)C)=O)CCC2(CCC2NC(=O)C(F)OC(F)(F)F)CC1 C1(CCC)CN(C(=O)CCCCOC)CCN1C(=O)C(O)CCSC N1(Cc2n(CCC)ccn2)CCN(C(C2CC23CC3)=O)CC1 N1(C(CC#N)=O)CC(NC(=O)CCCF)CC2(CCOCC2)C1 c1(CC)ccc(C(N2CCOC(CN(C(=O)CS(=O)(=O)N(C)C)C)C2)=O)c(N)c1 C1(O)(C(C)NC(c2c(CC)cns2)=O)CCN(C(C2CCCO2)=O)CC1 CC1(CCNC(=O)Cc2ccns2)CCN(C(C2(C#N)CCOC2)=O)C1 N1(C(c2cnc(C#N)s2)=O)CC2CC1CCC2NC(=O)CS(=O)(=O)CCO CCCC(CC)C(=O)N1CCCCC(CNC(c2cn(C3CCOC3)cn2)=O)C1 C#CC1(O)CCN(C(C2CC23CCN(C(c2cnnn2CC)=O)C3)=O)C1 c1(C(N2CCN(CC(=O)NCC(C)(F)F)C(=O)C2)=O)sc2ccccc2c1Cl C1(CC)CN(C(=O)CSCc2cccnc2)CCN1C(=O)C1=C(C)OCC1 c1(CC)nn(C)c(NCCCNC2CCCN(C(=O)CC3CSC3)C2)c1[N+](=O)[O-] c1(C(N2CC3CN(C(c4cnc[nH]4)=O)CC3C2)=O)ccc2c(Br)c[nH]c2c1 C1(CNC(c2cnns2)=O)CN(C(=O)C(F)(F)C(O)C2CC2)CC2(CCC2)O1 n1(CC(=O)NC2C(OC)CN(C(CN(CCC)C)=O)C2)cccc([N+](=O)[O-])c1=O C1(C2CCC2)(C(N2CCCC(C)C2CNC(=O)CCS(C)(=O)=O)=O)CC1(F)F N1(CC(=O)NCC=CCNC(C2CCC(C)(C)C2)=O)CCc2ccccc21 CC(c1ccccc1F)=CC(=O)NCC(CO)NC(=O)CC1CCCC(=O)N1 N1(C(c2c(C)c[nH]n2)=O)CCCC(C)(C)C1C(=O)N(C1CC(C(N)=O)C1)C C(C(N=c1ncnc2[nH][nH]c(C)c1-2)C1CC1)NC(C1N(C(CCC)=O)CCC1)=O N#CC1(C(N2CCC2CNC(=O)CN2CCC2)=O)CC(=O)C1 c1(OC)ccc(C=CC(N2CCOC(CS(C)(=N)=O)C2)=O)cc1C c1(CNC2CCC(NC(CCc3cccc(C)c3)=O)C2)ccc(C#N)cc1C N1(C(CCC)=O)CCC(N(C(C23CCC2C3)=O)Cc2ccccn2)CC1 C1(C(N2CC(OC)(CNC(=O)Cn3cccn3)C2)=O)CCCN(C(N)=O)C1 Cc1cc(C)c(C(=O)NCCN(C)C(c2cnn(C)c2Cc2ccccc2)=O)o1 C(=O)(C(F)C(C)(F)F)NC1(CCCC(=O)NC(c2cnccn2)(C)C)CC1 c1(SCCC)ccc(C(=O)NCC(C2CCOC2)NC(C2(CC)COC2)=O)cc1 CC(C)C(C(=O)NCCC(C)(C)CNC(c1ccoc1C1CC1)=O)N(C)C Cn1cc(N)c(C(N2CCN(C3CN(C(=O)C=CC4CCC4)C3)CC2)=O)n1 C1(NC(c2cccc(-n3cnnn3)c2)C)CCC2(CCN2)CC1 c1(C(=O)NCC2CC(NC(=O)C=CBr)C2)ncnc2c1CCCC2 C(C(C)(O)CC(=O)N1C(C(=O)NC(CO)CCCO)CC2CC12)OC C(=O)(C1=CCOCC1)N(CCC(C)NC(c1ccc(C(C)=O)nn1)=O)C CC(C)(CC(F)F)C(=O)NCCNC(c1ccccc1NCC(N)=O)=O N1(C(C2C(CCOC)C2)=O)CCOCC1(C)c1cn(CC2CC2)nn1 c1(C(=O)NCCN(c2ccnc(CC(C)C)n2)CCOC)cc2c(s1)CCOC2 N1(CC(=O)NC(C(C)NC(C2CC(C(=O)OC)C2)=O)CO)CC2CCC1C2 N1(C(C2(CC=C)CC2)=O)CCCCC(CNC(C2CC3(CCCC3)C2)=O)C1 CCC1=C(C(=O)N2CC(C3CN(C(c4cnn(C5CCC5)c4)=O)C3)C2)CCCO1 N1(C(CC2CC(CC)C2)=O)CC(C(=O)N(CCS(N)(=O)=O)C)(CC)C1 c1(C(N2CC(CNC(=O)CC3CC4(COC4)C3)OCC2)=O)nsc2ccccc12 c1(CC)ccc(F)c(C(=O)NCCN2CCN(C(C3CC3C3CC3)=O)CC2)c1F C1(NC(CC(C)(C)SC)=O)CC2CCC1N(C(C1(NC(C)=O)CCCC1)=O)C2 CC(C)(C)CCC(=O)NC1CCCC(NC(C2CC23CCOCC3)=O)C1 C(CC(C(=O)N1CC(O)CC1CNC(c1c(Cl)n[nH]c1C)=O)NC(N)=O)SC Cc1ccc(C(=O)NC(CNC(C2CCCCCC2)=O)C2CC2)c(C(C)C)n1 C1(OC)CC(NC(c2cnc(O)n2C)=O)CN(C(c2ccnn2CCF)=O)C1 c1(CN(CC(COC)C(F)(F)F)C)cc([N+](=O)[O-])c(C)cc1C C1(C)(CCNC(C(CC)C)=O)CCN(C(=O)COC(F)(F)F)C1 C#CC1(C(=O)NCCC2CCOC2)CCN(C(c2cccc(O)c2F)=O)C1 CCC1=NOC(C(N2CCC(C(C)NC(c3n[nH]cc3F)=O)CC2)=O)C1 c12cccc(OC)c1OCC(=O)NCCC2.C(=O)(CNC1C(=C)C1)N(CC)C c1(C(N(CCNC(=O)COCc2ccncc2)CC)=O)cc(C)c(F)cc1Cl Cc1cccc2cc(C(=O)NCC3CCN3C(c3cnn(C)c3F)=O)nnc12 c1(CC)nc(C(=O)NCC(CC)NC(c2cnoc2-c2cnn(C)c2)=O)co1 C1(C(=O)NCC2(NC(C(=O)NC(C)C)=O)CCOCC2)CCCS(=O)(=O)C1 C(c1cccc(Br)c1)=CC(=O)NC1CC(N(C(=O)CCCC#N)C)C1 C(=O)(C(O)CCn1cncn1)NC(C(CO)NC(CCC=CCC=C)=O)C CC(CC(=O)NC(C1(O)CN(C(C2(O)CCOC2)=O)C1)C)CC(F)(F)F N1(C(C(CC)OC)=O)CCC(NC(c2ccn(C)c(=O)c2)=O)C(C)(C)C1 Cc1ccc(Cl)c(OCC(=O)NCCC(C)NC(C2CN3CCN2CC3)=O)c1 N1(C(C(C(C)(C)C)=O)=O)CCN(C(=O)C=Cc2ccco2)CC(O)C1 C12C(C1(C)C)C(=O)NC2.C1(N(C)CC)CC(CC(=O)NC2(C3CC3)CCC2)C1 CC(CCNC(=O)Cn1cnc(C(F)(F)F)n1)CCNC(c1cccnc1N)=O C=C(C)CC(C(=O)NC1C(O)C2CCOC12)NC(C1CC=CCC1C)=O C(=O)(CC(C)C(=O)NC1CC(CC(=O)NC(c2nnc(O)n2C)C)C1)OC N1(C(c2n(C(c3ccccc3)C)ccc2)=O)CCN(CCO)C(=O)C1 C1(C)(CNC(C2C(CC(C)(C)C)C2)=O)CCN(C(c2cccc(C3CC3)c2)=O)C1 Cc1nc2cc(C(N3CC(C)CN(C(=O)C(C)C#N)C(C)C3)=O)cnc2[nH]1 c1(C(=O)NCC(C2CCC(=O)N2)C)ccc(Cn2cc(C3(C)CC3)nn2)cc1 c1(C(=O)NCCCC(C)NC(CCc2cc(C)no2)=O)ccc(C#N)nc1O c1(CC)occ(C)c1C(N1CCCCC1CNC(=O)CCCOC)=O C1(OC)CN(C(c2ccnn2CCF)=O)CCC1NC(=O)C(C1CCC(=O)N1)C c1(CC=C)cccc(CNC2CC(F)CN(C(C3CC3C)=O)C2)c1O C1(C2CCN(C)CC2)(C(N2CC3(CN(C(c4c(C)cc[nH]4)=O)C3)C2)=O)CC1 c1(C(N2CCC(C(C)NC(c3cc(C)[nH]c3)=O)CC2)=O)onc2ccccc12 N1(C(c2cc(Br)cs2)C(=O)OC(C)(C)C)CCN(C(C)CNC(=O)C2CC2)CC1 Cc1nn(C)cc1C(C)NC(=O)NCC1CC(F)(F)C1 C(=O)(CCS(C)(=O)=O)NC(CNC(C(CC#C)C1CC1)=O)(C)C1CCC1 C1(C(N2C(C)CC(O)CC2)=O)CCN(C(=O)CSC(F)F)C(C)(C)C1 c1(C(=O)NCCCC(C(=O)NC(CCOC)(C)C)O)ccc2nccn2c1 c1(C(=O)NC2C(C(N(C(C(N)=O)C3CC3)C)=O)OCC2)cccc(O)c1F C(CC)(C(=O)NC(CO)C(=O)NC1CN(C(=O)C2CC2)C1)=CCCC c1(C(N2CCC(C(C(C)C)NC(C(C)SC(C)C)=O)CC2)=O)cccc(Cl)c1F C1(CNC(C2C3CCC(=O)C32)=O)C(C2CC2)CCN1c1nnc(O)s1 c1(C(=O)NCCCNC(C(C)CN2CCOCC2)=O)nc(F)ccc1Cl Cn1cnc2c[nH]c(=NCC3(C)CCN(C(c4n[nH]cc4[N+](=O)[O-])=O)C3)nc12 c1(CNC(C2=C(C)OCCS2)=O)c(OC(F)F)ccc2ccccc12 CC1(C)CCC(NC(=O)C=Cc2nccs2)C(CNC(c2cc[n+]([O-])cc2)=O)C1 CCCCC(CC)C(=O)NCCCCN(C)C(c1cc(-c2ccccc2)no1)=O c1(CC)ccc(C)c(C(=O)N(CCCNC(C2C3COCC23)=O)C2CC2)c1 C1(NC(c2c(C)snc2)=O)CCC(C)(CNC(=O)CCC(=O)N(C)C)CC1 C(=O)(CC(C)(C)COC)N(C1CCN(C(=O)C(O)CCSC)C1)CCC C1(NC(CC2C(CC)C2)=O)CN(C(c2cc(C)nn2C(F)F)=O)CC12CC2 N1(C(CSCCC)=O)CC(OC)CC(NC(=O)C(C)Cc2ccc(C)cc2)C1 O=S(=O)(c1ccc(NC2CCC(CO)CC2)cc1Br)NC1CC1C1CCC1 N1(C(c2c(C)occ2)=O)CCC(O)(CNC(=O)C(O)C(F)F)CC1 Cn1ccc(=O)c(C(=O)NCC(C2CCCN2C(=O)CSc2cn[nH]c2)(C)C)c1 C(=O)(CC1c2ccccc2Oc2ccccc21)NC(CC)C N1(C(c2cc(OC)ncn2)=O)CCOCC(NC(=O)C(F)C(F)(F)F)C1 C12(C(N3CC(OC)C(NC(C4CC(C)(C)C4)=O)C3)=O)CC(N=[N+]=[N-])C1C2 O=C(C1NCCOc2cc(Br)ccc21)NCc1ocnc1C(F)F c1(NC(c2ccccc2S)=O)ccc(N=c2nc[nH]n3cc(Br)cc23)nc1 C1(C(=O)NCC2(F)COCCN(C(C3CCCO3)=O)C2)CCC(C2CCC2)CC1 C1(COC)CCCCN1C(C1CN(C(=O)Cc2c(C)n[nH]c2C)CCN1)=O CCCC(C)(C)CC(=O)NCC1CCC(NC(=O)CNC(c2cscn2)=O)C1 N1(C(c2nnn(CC)c2C)=O)CCN(C(C2CC23CC3)=O)C(CO)C1 N1(C(C(CCC)C(C)C)=O)CCC2(C=C(C(=O)N3CCCOCC3)C2)C1 C12(C(=O)NC(c3cccnc3O)C)C(NC(=O)Cc3cncnc3)C3CC1C2C3 C(CNC(c1ccc(CO)cc1)=O)(C(C)(C)C)NC(C(C1CCCC1)OC)=O C1(OC)CN(C(C2(F)CN(C(c3cc(C(N)=O)c[nH]3)=O)C2)=O)CC12CC2 Cc1cc(C)c(NC(C2CN(C(c3cc(C)c(F)cc3Br)=O)CCS2)=O)c(Br)n1 c1(CC(=O)NC(C2CCN(C(=O)CCNC(=O)CO)C2)C)occc1C(=O)O C(=O)(C(O)CCN(C)C)NC1(C(N(CCCC(=O)OC)C)=O)CCCC1 CC(C(=O)NCc1nnc(C2CC2)o1)S(=O)(=O)Cc1ccc(C#N)cc1 c1(CCC(=O)NCC2N(C(C(N)=O)=O)CC(O)C2O)cncc2ccccc12 Cc1ccc(CCC(N2CCOCC2CNC(=O)C(C)CC2CCC2)=O)cc1 c1(C(=O)NCC(CNC(c2c(F)ccc(CC)c2)=O)O)ccc(OC)c(F)c1F Cc1[nH]nc(-c2nc(CC(F)(F)F)nn2-c2ccnc(F)c2)c1C CCC(C)CC(=O)C(=O)NCC1CN(C(=O)CCCc2ccsc2)C2(CCC2)C1 N1(C(c2c(CC=C)cccc2)=O)CCN(C)C(C(=O)NC(C2CSC2)C)C1 C=CC(C)(O)CC(=O)NCCC1CCCN(C(c2ccc(CC(N)=O)cc2)=O)C1 Cc1ccc(C(=O)NC2CC2NC(c2ncsc2C(F)(F)F)=O)c(C)c1 N1(C(c2cc(C)[nH]c2)=O)CCc2c(C(N3CCC(N4CCC4)CC3)=O)csc2C1 N1(C(C2(CSC)CC2)=O)CC(NC(=O)CC2CC2)C(N=[N+]=[N-])C1 C=CCN=c1[nH]cc(C(=O)NC(C)CCNC(c2cnc(C(F)(F)F)s2)=O)s1 Cc1ncnc(C)c1CC(N1CCC(CNC(=O)C(N)=O)C(C)C1)=O Cc1cccc(C(=O)NC2CN(C(=O)C(F)CC3CCC3)CC2O)c1 N1(CC(=O)NC2(CF)CCN(C(=O)CCNC(C3CCC3)=O)C2)CCCCC1=O CCC(CC1CCCC1)C(=O)N1CCC(F)(CNC(c2ncccc2SC)=O)C1 C1(OC)(CNC(=O)COC2CCN(C(=O)C=Cc3cscn3)C2)CCOC1 Cc1c(NC(=O)NNC(=O)c2ccon2)cccc1Br c1(C(=O)NC2CC(C(N(CC(N)=O)CC)=O)CC2O)ncc2ccccn12 c1(C(C(=O)NC2CCOC2)N(CC(C)(C)C)CC)ccc(C)c(Br)c1 S(=O)(=O)(c1ccc(OCC(=O)O)cc1)NCCN1C(CC(=O)O)CCC1 N1(C(c2cnc(COC)s2)=O)CCC(C)(NC(c2csc(C)n2)=O)C1 c1(-c2cn(CC(=O)NC(Cc3ccccc3)C3CC3)nn2)cnccc1Cl c1(C(=O)NCC2C(NC(C(CC)NC(C)=O)=O)CC2)ccc(C)cc1N n1(CC)nc(C(N2CCOC(C(C)NC(c3ccc(C(N)=O)[nH]3)=O)C2)=O)cc1C C(=O)(C(CO)C(F)(F)F)N1CC(C)C(NC(C2(C)CC3(CC(=O)C3)C2)=O)C1 c1(N2CC(O)(CCNC(c3cc(C)n(C(C)C)n3)=O)C2)ccnc2ncnn12 c1(C(=O)NCCOCCNC(c2cc(Cl)ccn2)=O)cc(=O)c(Br)c[nH]1 C1(NC(C=CCOC)=O)CN(C(=O)CC(c2cccc(F)c2)O)C(C)(C)C1 N1(C(C=CC=CC)=O)CC2C=CC1C(C(=O)NC1CCC(O)CC1)C2 C1(COC)CC(CNC(C2SCCCS2)=O)N(C(=O)C(c2ccn(C)c2)C)C1 C(CCF)(C(=O)Nn1nnc2c1CCCC2)NC(CCSCCCC)=O Cn1nc(C(N2CCC(CNC(C3CC4(C3)CC4(F)F)=O)C23CC3)=O)c(Cl)c1Cl c1(C(N2C3C(NC(c4ccc(CC)o4)=O)CC(C3)C2)=O)nccn2ccnc12 CC(c1cccnc1)=CC(=O)NCC1CC(O)CN1C(=O)CC1CNC(=O)C1 CCC(CC(=O)NC1CCN(CCCO)C1)NC(=O)C=Cc1cnn(C)c1 CC(CC(C)(C)C)NC(C1CCC(C(C)(C)O)CC1)=O C(c1ccccc1)=CC=CC(=O)NCCCC(C)NC(CC=CCC)=O Cc1cc(C(=O)NCCCN(C(C2(CC(F)(F)F)CC2)=O)C2CC2)oc1C C1(OC)CCC(CC(=O)N(CCNC(C2CN(C3CC3F)C2)=O)C2CC2)CC1 c1(C(=O)NC(CC(=O)N2CC(C(CC)CC)C2)COC)cc2ccccn2c1 c1(OCC)nc(C)ccc1C(=O)NCC(C)(O)CNC(=O)CCCn1ccnn1 N1(C(C2N(C(C(C(C(C)C)OC)O)=O)CC(C)CC2)=O)CC2(CCCCCC2)C1 CC1CN(C(C23CC2CCN3C(C2COCCN2C)=O)=O)Cc2c[nH]nc21 CN1CCC(C(=O)NC2(CNC(=O)CCCF)CCOCC2)CC1 c1(C(C)C)cc(C(=O)NCC2CC2NC(=O)CCc2cnccn2)n(C)n1 C(C(=O)NNc1ccc(F)c(Cl)c1)C1C(C(C)C)CCCC1 CCC(C)CCCC(=O)NCC#CCNC(c1ocnc1C1CC1)=O C(c1c(Cl)nc2ccccn12)=CC(N1CC2C(CNC(C3(F)C(C)C3)=O)C2C1)=O CC1C(NC(=O)CC(C)C2CC2)CCCN1C(=O)Cc1nc(C(C)(C)C)cs1 Cc1ccc(Br)c(OS(=O)(=O)CC2CC2(Cl)Cl)c1F C=CC1(C(=O)N(C)CCC2CCCC2)CCN(C(=O)C(C)CC=CCC)CC1 C1(NC(CCC2(C)CCC(=O)N2)=O)C2CC1CN(C(C1CCC(F)(F)C1)=O)C2 CC1(C)CC(C(N2CC(NC(=O)CN3CSCC3=O)C2)=O)CCO1 C1(C2CCOCC2)(C(=O)NCC2(C)CCN(C(c3ccsc3Cl)=O)C2)CC1 S(=O)(=O)(c1ccc(=NCc2ccc(Br)s2)[nH]c1)NCCn1c(C)nnc1 C1(C(=O)NC2CC(CCNC(=O)C(O)c3ccsc3)C2)(OC)CCSC1 Cc1cccnc1C(F)(F)C(=O)NC1CN(C(=O)C(C)OCC(C)C)CC1C c1(C(N2C(C(C)NC(C(C)C)=O)CCC2)=O)cc([N+](=O)[O-])c[nH]1 c1(N2C(C(N(CC(=O)Nc3ccsc3)CC)=O)C(C)CC2)nnccc1C#N C1(CNC(C2CC2C2CC2)=O)CCCCN1C(=O)CCC=CBr c1(C(=O)NCC(C2CC2)NC(C2C(C(=O)OCC)CC2)=O)cnc(CC)nc1O C(C(CNC(C1CC(=O)N(C2CC2)C1)=O)S(C)(=O)=O)NC(c1c(C)cno1)=O C#CC1CCCN(C(c2ccnc(F)c2C)C(=O)NCC=C)CC1 C1(C(=O)NCCC2CC(C(=O)NCC(C(=O)OC)(F)F)C2)CC2C=CC1CC2 c1(N(CC)CC2CCOC2)nnc(-c2cc(-c3ccncc3)[nH]n2)n1C CCC(CCC(=O)NCC(C)(O)C1CCCC1)NC(c1nnn(C)c1C)=O N(C(=NCc1ccc(C)o1)NC1CCCCC1)C(C#C)C(C)OC c1(C(=O)NCC2CCN(C(C(CC)(C)CC)=O)CC2)cc(OC)c(OC)cc1O N1(C(C=CC)=O)CCC(C2CC2)C1C(=O)N(CC(C)(C)C(=O)NC)C1CC1 N1(C(Cc2c(C)n[nH]c2)=O)CC(C(=O)NCCc2cnnn2C)C(F)(F)C1 C(=O)(C1=NOC2(CCOC2)C1)NCC1CN(C(C(n2ccnn2)C)=O)C(C)(C)C1 CCC(C)CC(C(=O)N1CC2CCC1CC2)NC(c1ncc[nH]1)=O c1(NCC(c2cc(OC)cc(OC)c2)O)cnn2c1OCC(N)C2 N1(C(=O)N(c2ccc(F)cc2)CCO)CC2(CCCC2)c2c(F)cccc21 CC1COCC(CC(N2CCC(CC(=O)N(C3CCCCC3C)C)CC2)=O)O1 CCCC(CC)C(=O)N(CCCNC(C1CC(n2cccn2)C1)=O)C(C)C C1(OC)CC(CNC(c2cc(F)n(C)n2)=O)N(C(=O)CNC(=O)CN(C)C)C1 N1(C(C2CCC(C)(C)OC2)=O)CC2(CCN(C(c3cc(CCO)on3)=O)C2)C1 c1(C(=O)NCC2(NC(=O)C#CC3CCC3)C(C)CCCC2)ccc2nsnc2c1 c1(OC)ccc(CC(N2C3CCC2C(NC(c2cccc(Cl)c2)=O)C3)=O)cc1F C=CCC(C(=O)N(CCCC(=O)NC(C(C)C)c1nc[nH]n1)C)OC C(CNC(=O)C(C)(C)CC1CCC1)(CC(C)C)NC(COCC#C)=O c1(C(=O)NCC(C2N(C(CC=C)=O)CCC2)(C)C)c(C)cc(=O)oc1C C(=O)(C(C)C1=CCCC1)N(CCCCN(C(c1c(C#C)c[nH]n1)=O)C)C N1(C(C2(C)N(C(C(CC)SC)=O)CC=C2)=O)CCOC(C)(C)C1C N1(C(CN2CC(CC)C2)=O)CCOCC(NC(=O)Cc2c[nH]nc2C)C1 CC(CN=c1nc2c(cnn2C)c(NCCc2n[nH]c(C3CC3)n2)[nH]1)S(C)=O CC(O)CCCC(=O)NC1CCCN(C(=O)C(C(C)(C)C)N2CCCCC2=O)C1 N1(C(C(C)C2CCCCC2)C(=O)Nc2ccccc2)CCCC2(CNC(=O)O2)C1 C#Cc1c[nH]nc1C(=O)NCCCCN(C(=O)CCCNC(=O)C1CC1)C N1(C(C)=O)CCCC(O)(CC(=O)NCC(C)(C)NCc2nccc(C)n2)C1 CCCCCC(C)CC(=O)NCC(=O)NCCOCCOCc1nc(CC)no1 c1(CC(N2C(CNC(C(C)OCC)=O)(COC)CCC2)=O)cnn2ccccc12 N1(C(CC=C)=O)CC2(C1)OC1(C(C)C)CC2(NC(c2ccc(CSC)o2)=O)C1 c1(NC(C(=O)NC(CC)C(O)c2ccccc2)=O)ccc(OC)nc1Br c1(C(=O)NCC2C(NC(c3sc(CC)c(C)c3)=O)CC2)cc(S(C)(=O)=O)c(C)o1 C(=O)(CN(C)N1CCCc2c1c(N(C)CC(=O)OC)nn2C)NC c1(C(=O)NC(C)C(CO)NC(=O)C=Cc2ccc(O)cc2)ccn2c1CSCC2 N1(C(C2CN(C(C)C)C(=O)CC2)=O)CC(NC(=O)CNS(C)(=O)=O)CC2(CC2)C1 Cc1cc(OCCC(=O)NC2CC3CCC2N3C(=O)C(C)(C)CO)c(C)c(C)c1 CCCCCCC(C)C(=O)OCC1CCC(Nc2ncccc2Cl)CO1 Cc1[nH]nc2ncc(C(=O)NCCCC(C)NC(c3cc(Cl)c(Cl)n3C)=O)cc12 C1(C(N(C2(C(=O)NC(c3ccsc3)C)CC2)C)=O)CCCSC1 c1(C(N2CC(NC(C(C(C)C)NC(C)=O)=O)C2)=O)cccc(N=[N+]=[N-])c1 C1(NC(CC(C)c2ccco2)=O)COC2(C1)CN(C(c1ccc(F)c(O)c1)=O)C2 C1(C)(CC)CN(C(C2(CC)CCN(C(c3cc(OC)nn3C)=O)C2)=O)CCO1 Cc1nc(C(=O)NC2CC3(C2)CC3NC(=O)CCc2ccccn2)c(C)s1 C(=O)(CCC(C)C)NCC(=O)NC(CNC(c1c(C)nn[nH]1)=O)C1CCC1 CCC(CC(F)(F)F)C(=O)N1CCC(NC(c2nc(Cl)cs2)=O)C(O)C1 c1(NCc2snc(C)n2)nc2ccccc2nc1NCC1OCCc2sccc21 C1(CC)(CC)CCCN(C(C(=O)NC2CC(F)(F)C2)c2cn[nH]c2)CC1 C(c1ccc[nH]1)=CC(=O)NCCCOCCN(C(C1N(CC)CC1)=O)C C(=O)(CCCCCC1CC1)N(C1CCCCC1NC(C1(C)CCCNC1=O)=O)C C#CCC(C(=O)N(CCNC(C1(CCF)CC1)=O)CC1CC1)C1CC1 N1(C(C(=O)NC(CC)C)C(C)C2CCCCC2)CCCN(CC(O)CO)CC1 N1(C(C(=O)Nc2cn(CCOC)nn2)=O)CCC(C(C)NS(C)(=O)=O)CC1 C1(CNC(=O)COC2CCCC2)CCCN(C(c2ccc(F)cc2)=O)CC1 C12(C(N(C)CC3CCCCO3)=O)COCC1CN(C(c1ccccc1O)=O)C2 C(=O)(CCS(=O)(=O)c1ccccc1)N1C(CS(=O)(=O)NC)CCCC1.C(=O)C(C)C c1(C(=O)NC2(CCNC(=O)CCc3cccnc3)CCCC2)cc(CO)ccn1 N1(C(COC2(C)CN(C(c3ccc(C)nc3O)=O)C2)=O)CCc2c[nH]nc2C1 N1(C(C(n2c(C)ncc2)C)=O)CCC(C)N(C(=O)CC=C(Cl)Cl)CC1 Cc1nc(CCC(=O)NC(C)C(CO)NC(C2COC(=O)O2)=O)[nH]c1C Cc1cc(C(=O)NCC2CC2NC(c2cnc(Cl)c(N)c2)=O)ncc1C(N)=O S(=O)(=O)(c1c[nH]ccc1=NCC(O)C(N)=O)NC(CCS(C)(=O)=O)c1ccccc1 C(=O)(C1CN(c2ccccc2)c2ccccc21)N1CCCC(n2ccc(CO)n2)C1 c1(C(=O)Sc2n(CCC)ncc2C(=O)OC(C)C)ncc(Cl)c(SC)n1 c1(C(=O)NCC2N(C(=O)C3=NNC(=O)C3)CCN(C)C2)c2c(nn1C)CCC2 N1(C(C(N2CCC(O)CC2)C)=O)CCC(C)C(CNC(c2nccn2C)=O)C1 N1(C(C2(C)CCC2)=O)CCN(CC2CCCN(C(C3(CO)COC3)=O)C2)CC1 Cc1nn(C)c2c(NCC3CCCOC3)nc(N3CCC(C(C)C)(CO)C3)nc12 c1(C(C)C)nc(=NCC2C3CN(C(C4(C)CCCN(C)C4)=O)CC23)s[nH]1 Cc1cn2cc(C(=O)NC3(C)CCN(C(C4(n5cncn5)CC4)=O)CC3)nc2s1 C(CCCC(=O)NC(C)(C)CNC(=O)Cn1cnc(C(=O)OC)c1)OC Cc1ncc(Br)c(N(C2CC(N)C2)Cc2cc[nH]c2)n1 c1(C(=O)NCc2cc(C(=O)NCc3cc(C)no3)sc2)c[nH]c2nccc-2c1.C C1(CC(N2CC(CNC(C(CC)NC(C)=O)=O)OCC2)=O)(CC)CC(F)(F)C1 c1(C(=O)NCC(=C)CCNC(c2[nH]nnc2C)=O)cnc(O)cc1O O=C(CCC1=NNC(=O)CC1)NCC1CCCCN1C(=O)CCN1CCOCC1 C1(CN(C(C=COCC)=O)C)CN(C(C2CCS(=O)(=O)C2)=O)CCO1 N1(C(C(CC=CC)CC)=O)CCCC(C)(C)C1CNC(=O)CNC(C)=O C1(C(=O)NC(c2nc(C(=O)N(CC(Cl)Cl)C)co2)C)CCCC(C#N)C1 C(=O)(C#CC(C)(C)C)N(C1(C(N2CC(C#C)C2)=O)CC1)C Cc1ccc(CC(N2CCCC(C(C)NC(c3cscn3)=O)C2)=O)c(Cl)c1 C(=O)(C(C(C)(C)C)Nc1csc(CC)n1)NCC1CCN(CCC)C1 CC(C)CCCC(=O)NC1CCCCN(C(c2ccc(F)cc2N)=O)C1 CC1CCC(C)C1NC(=O)CCC1CCN(C(=O)CC2(O)CCCOC2)CC1 N1(C(c2c(C)nsc2N)=O)CCC2(CCC(NC(C3(C(N)=O)CC3)=O)C2)CC1 C1(CNC(=O)CNc2ccccn2)COC2(CCNC2)C1 c1(C(=O)NC2C(C)CN(C(c3ccon3)=O)CC2)ccc([N+](=O)[O-])c(N(C)C)c1 N1(C(CC(C)SC)=O)CCC(N(C(=O)C2=CCCS2)CC2CCCO2)CC1 CN=c1[nH]c(=NCCc2cccc(F)c2)[nH]c(=NC2CN(C)C3(CCCC3)C2)[nH]1 C1(NC(c2ncn(CC)n2)=O)CCCC(NC(=O)CSc2ccccc2O)C1 c1(C(=O)NCCCC(C)NC(Cc2c(C)ccnc2)=O)ccc2c(O)n[nH]c2c1 C1(OC)CC2(C1)CC(NC(=O)CC1CC(NC(=O)C(F)(F)C(F)F)C1(C)C)C2 Cc1ncc2n1CC(C(N1CC(CNC(=O)CCC3CC3)C(C)(C)C1)=O)CC2 C1(C(=O)NCC2(C(=O)NCC(O)COCC)CC(=C)C2)CCCCN1C N1(C(CC2C=NN(C)C2=O)=O)CCC(C(N2CC3CCC(C2)N3C)=O)C(C)(C)C1 C1(NC(C(COC)NC(c2ccncc2F)=O)=O)CC2CC1CC2(C)O O=C(CC(=O)N1CC(O)(CNC(C2CN(C3COC3)C2)=O)C1)NCC1CC1 C(=O)(C#CC(C)(C)O)NC(C)C(C)C(=O)N(C)CC1(CO)CC1 N=c1ccc(C(=O)NC2CC(NC(c3cncc(Cl)c3)=O)C2)c[nH]1 C(=O)(CCCS(C)(=O)=O)NC(C1CCCC1)CNC(C1CCC(C)CC1)=O Cc1ccc(O)cc1C(=O)N(C1(C(=O)N(CC(O)C(C)(C)C)C)CCC1)C1CC1 C1(NC(c2c(C)nns2)=O)COCCN(C(C23CC(CO)(C2)OC3C)=O)C1 C1(C)(CN(C(C(C)OCCOC)=O)C)CCCC1NC(c1cocn1)=O C(C(C)(C)C#CC(=O)N(C)CCc1ncon1)NC(C1C(C)CCOC1)=O CCC(C)C(=O)NNC(=O)NCCc1ccc(C)cc1F C12(C(=O)NC3CN(C(CC(C)n4cccn4)=O)C3)CCC(C1)C(C)(C)O2 C1(F)(CNC(c2c(C)cc(C)s2)=O)CCC(CNC(C23CCCC2C3)=O)CC1 Cc1cc(NC2CCN(C(=O)CSc3ccc(F)c(F)c3)C2)n2ncnc2n1 c1(C(=O)NCCNS(CC)(=O)=O)cccc(NC(=O)C(F)Cl)c1 C1(CNC(C(C)SC(C)C)=O)(CNC(=O)Cc2cocn2)CCCCC1 C1(C(=O)NCCN(C(C2(O)CCCCCC2)=O)C2CC2)CCCC2CCCN12 Cc1c(Br)sc(C(=O)NC2CCC(C)(C(=O)O)C2)c1Br Cc1nc(NCC(C)(C)NC(c2ccsc2)=O)ncc1[N+](=O)[O-] C(CN=c1[nH]c(=NCc2cocn2)c2[nH]ccc2[nH]1)C1CC(C)OCC1 c1(C(N2C(C3CCN(C(c4cnns4)=O)C3)CCCC2)=O)ccc(Cl)c(F)c1F N1(C(CC(C=C)CC)=O)CCC2(CC1)CC2C(=O)NCC1(C2CC2)CCC1 Cc1c(C(=O)NCCCNC(=O)C2=COCCC2)cc(C(F)(F)F)cc1N c1(CN2CC(NC(c3ccc(OCC)nc3)=O)C(F)C2)ccc(I)c(F)c1 CC1COCCN(C(C2CCN(C(=O)CSc3nc[nH]n3)C2(C)C)=O)C1 N1(C(C(CC=C)C(=C)C)=O)CCC2(CC1)CC(C(=O)NCC(=O)N(C)C)CO2 Cc1cc(C(N2CCCCC2CCNC(c2cnco2)=O)=O)c2c(c1)CCCN2 C1(CC)CN(C(=O)COc2cc(C)on2)CCC1NC(c1cn[nH]c1)=O C#CC1(C(N2CC(N(C)C)C(C)C2)=O)CN(C(c2ccc[nH]2)=O)C1 C(C1c2ccsc2CCN1C(=O)C=CC1CCOC1)NC(Cc1scc(C)c1)=O Nc1cc(C(N2CC3C(CNC(c4ccc(F)s4)=O)C3C2)=O)cc(N)c1 C(=O)(CN=S(C)(C)=O)N(CCCCN(C(CCC(=O)OCC)=O)C)C CCCCC(C)C(C)(c1nnnn1C(C)C)NCc1ccc(Br)nc1Cl C1(C(N2CCC(NC(C(CCOC)C)=O)(COC)C2)=O)CCc2ncc(C)n2C1 c1(CC)cn2c(n1)CCC(C(N1CC(C(C)NC(c3cnc(S)n3C)=O)C1)=O)C2 Cc1nn(CCCl)c(C)c1NC(N1CCN(c2ncccc2C(F)(F)F)CC1)=O Cc1ccc(Cl)c2[nH]c(C(=O)Nc3ncc(-c4ccc(F)cc4)s3)cc12 c1(C(=O)NCCC(C)NC(COCC=C)=O)cc(Br)cc(F)c1F C1(C(N(C)Cc2ccc(C)cn2)=O)N(C(C2CC2(Cl)Cl)=O)CCC1(C)C c1(N(C)C)cccnc1C(=O)NC1C2CN(C(C3(C(F)(F)F)CCCC3)=O)CC12 Cc1ccc2c(c1)SC(C(N1CC(NC(c3[nH]cc4c3CCS4(=O)=O)=O)C1)=O)C2 C(CCN=C(NCC1CCCCC1(F)F)NC1CC1)N(CCC)CC C(C(C(C)(C)C)NC(c1csc(C2CC2)n1)=O)NC(CN1CCC(C)C1)=O C1(CC(=O)NCCC(Cn2cc(CCCCC)nn2)(F)F)CCC2(C1)CC2(F)F c1(NC(C(C)NC2CCNCC2(C)C)=O)ccc2c(c1)OCO2 c1(NC(=O)NCCSCC)cccnc1SC(F)F c1(C(=O)NCc2cc(C(=O)NC(C)C(C)n3cncn3)no2)nccnc1N Cc1ccc(C(=O)NC(c2cnccn2)C)c(F)c1C c1(C(C(=O)NC)N(CC(=O)OCC)CC(C)C)cn(C(C)(C)C)nn1 N1(C(CN(C)C2CC2)=O)CCC(NC(c2cnn(C)c2Cl)=O)C1c1ccccc1 N1(c2nnc(SC)s2)CCC(CCCCCNC(=O)CC(C)(F)F)CC1 N1(C(C2CC(C)(C)OC2)=O)CCCCC(NC(=O)CCCC(=O)C2CC2)C1 C(=O)(CCS(=O)(=O)C1CCCC1)NCC1(C)CN(C(c2cc(F)c[nH]2)=O)CCO1 C12(CNC(NNC(c3c(=O)cc(C)[nH]c3)=O)=O)CCC(C#N)(CC1)CC2 c1(OC)ccc2c(c1)OCC2NC(=O)NCc1nc(C(F)(F)F)nn1C N1(C(C2CCN(C(CC)=O)C2)=O)CCCC(CCCNC(c2cc(O)cs2)=O)C1 N1(C=O)CCCN(C(=O)CNC(N)=O)C(C)C1.c1(OC)cc(C(F)(F)F)cc(OC)n1 C(N=c1nc(C)nc2[nH][nH]cc1-2)c1nc(N2CCCC(N(C(C)=O)CCO)C2)sc1 Nc1ccc(C(=O)N(C2CCN(C(C3C=CCCC3)=O)C2)CCO)cc1Cl Cc1cc(=NCC2CCC(NC(c3csnc3C)=O)C2)[nH]c(CC2CC2)n1 c1(C(N(CCNC(=O)CCc2cc(Cl)cs2)CC)=O)ccc(C#N)cc1 C1(C(N(CC=C)CC2CC2)=O)CC2CCC(C1)N2C(=O)Cn1ccccc1=O c1(CC(=O)NC23CC(NC(=O)CC4C=CCCC4)(C2)C3)cnc(C2CCOC2)s1 C1(CCNC(COCCCCC)=O)CN(C(=O)Cc2nnc(CC)o2)CC(C)O1 CC1(NC(=O)C(O)CCl)CCN(C(=O)NC2CC2c2cccc(Cl)c2)C1 Cc1c(C(=O)NCC(C)NC(=O)Cc2nnn(C(C)(C)C)n2)[nH]c2c1CCCC2 CCC(CC)CC(=O)N1CCN(C(c2cnn(C)c2Cl)=O)C(CCO)C1 N1(C(=O)Cc2cn3ccsc3n2)CC2CC1CCN2C(C1CC12CCCC2)=O C1(OC)CCCC(CC(=O)NCCC2CCCN2C(=O)C(O)Cc2cnc[nH]2)C1 C(C)(C(=O)N1CCC1CNC(=O)C(C)N(C)CCNC(C)=O)=C(CC)C N1(C(C=CCN(C)CC)=O)CCC2(CC1)CN(C(=O)C(O)C1CCCC1)C2 N1(C(CC2(C)CCCC2)=O)C2CC1CN(C(c1scnc1Cl)=O)C2 c1(C(=O)NC2(C)CC(NC(C(C)C(C)(F)F)=O)C2)cnn2c1OCCC2 Nc1c(F)ccc(F)c1C(=O)NCC1CCCN1C(C1(C(F)F)CCCCC1)=O C1(C(C)C)CN(C(c2ccc(Cl)s2)=O)CCC1NC(C1CC(C(N)=O)C1)=O C=CC(C)(CC)C(=O)N1CCCOC(CNC(C2(COC)CCCCO2)=O)C1 Cc1cc(C(=O)NC2CC2CNC(=O)CC2CC3(CC3)C2)c(C)cc1Cl C(=O)(C(N)CC(C)(C)O)NCc1ccc(C)nc1Cl C=CCC(CC=C)C(=O)N1CCCC(N(CCF)C(c2ccc(C)nc2C)=O)C1 n1(CC)nccc1C=CC(=O)N(C1CN(C(C2CC(CF)C2)=O)CC1O)C CC1CN(c2ccc(Cl)nn2)CC(C)N1Cc1ccc(-c2ccccc2)nc1 C1(C(N2CC(C(=O)OCC)C2)=O)N(C(c2cc(COC)no2)=O)CCC1(C)C C1(n2cc(C(C3CC3)OC)nn2)CC2CCC(C1)N2C(C1CC1(C)C)=O c1(CC(=O)NC2CCC(NC(C3(C(C)C)CC3)=O)C2)cncc2ccccc12 C#CC1CCCN1C(=O)C(CC=CC)NC(=O)C(C1CC1)C1CC1 CCCCCCC(C)C(=O)NC1CCC(NC(c2sc3nccn3c2C)=O)CC1 C1(C(=O)NC2C(NC(c3csc(-c4ccsc4)n3)=O)COC2)C2CC(F)(F)CC12 CC(C)(CCNC(=O)Cn1ccc(C2CC2)n1)NC(=O)COC1CCC1 N1(C(=O)COC2CCCC2)CC2CCC(C1)N2C(c1ncc2[nH]ncc2n1)=O CN1CCN(C(c2cc(F)cc(F)c2)=O)CC1CNC(=O)CCC1CC1 C(=O)(C(CCC)CC(C)C)N1CCC(OCCNC(C(C=C)(C)O)=O)CC1 c1(CC(=O)NC2C(NC(C3N(C)CCOC3)=O)CCC2)cc(F)ccc1O Cc1ccc(C(O)C(=O)NC2COCC2NC(=O)CCNC(N)=O)cc1 C1(N(c2ncc(F)cn2)C(c2cnn(C(F)F)c2)=O)CCCC12CCNCC2 c1(OC)c(C(=O)NCC2(CNC(C3CC3C#N)=O)CC23CCC3)ccc(Cl)c1Cl C(=O)(CCC(=O)C(C)(C)C)N1C(CC(N2CCC(C(C)C)CC2)=O)CCC1 c1(C(=O)NCC(C)(C(C)C)NC(C(CCCC)C)=O)cccc2c1C(=O)CCN2 C1(CC(=O)NCC2COC(CNC(=O)CN3CCSCC3)C2)CC(=O)NC(=O)C1 S(=O)(=O)(c1c[nH]ccc1=NC(C)c1cc2ccccc2s1)N1CCCCC(C)C1 C1(C(=O)NC(CCC)C(=O)NCC2CC3CCC2CC3)CCCCCN1C [N-]=[N+]=Nc1ccc(C(=O)NC2COCCN(C(C3CNC(=O)N3)=O)C2)cc1 CC1CCC(NC(=O)CCC(C)(C)C)CN1C(=O)Cn1cnnc1 C1(NC(c2cc(C)no2)=O)CCN(C(c2cccnc2-n2nccn2)=O)CC1O c1(C(N2CC(CCCCNC(c3cc(Cl)ncc3F)=O)C2)=O)ccc2cnoc2c1 C1(CNC(C2C(C)C(=O)C2)=O)(NC(=O)CC2CCOC2)CCCCCC1 CC(C)(C)S(=O)(=O)CC(=O)NCC1CCCN1C(=O)Cc1cnns1 C(N=c1nc2c(Br)csc2c[nH]1)C1C(NC(=O)CC(O)c2ccccc2)CCC1 N1(C(C2C(C3CN(C(C4CCSC4)=O)C3)C2)=O)CC2CCC1C(O)C2O c1(C(N2CCCCC(NC(C(CC)CC)=O)C2)=O)[nH]c2ccccc2c1C#N N1(C(Cc2c(C)cc(F)cc2)=O)C2CCC1CN(C(c1ccc(Cl)o1)=O)CC2 C1(C)(CC)CCC(C(=O)NCC(C2CCCCC2)NC(C2(OC(C)C)CC2)=O)O1 CC(CF)CC(=O)N1CC(F)CC1CNC(c1ccc(N2CCCCC2)cc1)=O N#Cc1cc(C(=O)NCC2CC2CNC(c2ccc(Cl)s2)=O)cc(F)c1F CC1CN(C(C2(C(F)(F)F)CC2)=O)CC(C)N(C(c2csc(S(C)(=O)=O)c2)=O)C1 N1(C(C=CC)=O)CCN(C(c2cc(C)c(Cl)c(N)c2)=O)CCC1C C(C(C)CC(=O)N1CCC(CN(C(=O)CCc2ccc[nH]2)C)C1)OC c1(C(=O)NCC2CCC(NC(c3nncc(C)c3)=O)C2)cncc2cnccc12 CCC(CC(=O)N1CCN(C(c2cnc(C(N)=O)s2)=O)CCC1C)CC(F)(F)F C1(NC(c2n(CC)nc(C)c2)=O)CCCN(C(c2ccc(C)cc2OC)=O)C1C C(C(=O)NC1(C(F)F)CCCC1)(C(C)C)NC(CCOCCOC)=O c1(C(=O)NC2C(NC(=O)CC3C=CS(=O)(=O)C3)CC2)ccc2c[nH]nc2n1 C1(COC)(NC(=O)CSC2CCOC2=O)CCN(C(C2CCS2(=O)=O)=O)CC1 c1(C(=O)NC2(CNC(c3c(Cl)cc(C)c(F)c3)=O)CC2)cc(F)c(F)c(F)c1F N1(C(CNC(N)=O)=O)CC2CCOC2(CNC(=O)CN2CCC(O)CC2)C1 C1(C)(C(N2CC(CNC(c3c(C)nc(=N)[nH]c3)=O)OCC2)=O)CCCCC1(F)F N1(C(C=CCCC=C(C)C)=O)CC=C(CCNC(C2CC2C)=O)CC1 C1(NC(c2cc3ncccc3[nH]2)=O)CC2CN(Cc3ccc(F)c(F)c3)CC2C1 C(C(C)(C)CC(=O)NCC(O)C(C)O)NC(c1cccc(CC)n1)=O C(CNC(C1CCC(C)O1)=O)(C(C)(C)C)NC(Cn1ncc(C)c1)=O C1(CC2CCC2)C(=O)N1.C(CC(=O)N1CCC1C1CCC1)NC(=O)OCC C(CCC(C)(C)C(=O)NCc1cccc(C#N)n1)NC(CCCCC=CC)=O Cc1cnc(C(=O)NCCCN(C(C2CCCC(C)(C)O2)=O)C(C)C)c(F)c1 N1(C(CSC)=O)CCC(C(=O)NC2C3CCC2CC3)C1C(C)C CN1CCN(c2ccc(CCNC3CCN(C4CC4)C3)cc2)CC1 CC1(C)C(=O)NCC1NC(N1CCC(O)(C(N)=O)C1)=O C1(CNC(C2C(CC)CCO2)=O)CCCC2CN(C(C3CCCCC3C)=O)CC12 c1(N(CC(F)Cl)C)ccc(S(=O)(=O)N2CC3CC3(CO)C2)cc1Cl C(CC(=O)NCc1cnn(C)c1OC)(C(F)F)NC(C(C(C)C)OCC)=O Nc1nccnc1C(=O)NCCCCNC(c1ccc(Cl)nc1)=O c1(-n2c(C)nnc2)ccc(C(=O)NC2CC(F)(CNC(c3cccs3)=O)C2)cc1 N1(C(c2nn(C)c(C(F)(F)F)c2)=O)CCCN(C(C2CCC3CC23)=O)CCC1 C=CC1(C(=O)NCCCCC2CCCN(C(=O)C(O)C(C)(C)C)C2)CCCCC1 c1(C(=O)NCc2ccncc2F)ccc(F)c2cnccc12 c1(CN2C(C(=O)Nc3nccc(F)c3F)CNCC2)c[nH]c2ccc(Br)cc12 C1(NC(C2CC(C(C)C)C2)=O)CCC(NC(=O)C(C)(C)Cl)C1 Cc1cc(Br)c(C)c2c1N(C(=O)CCOc1cccc(C(N)=O)c1)CCC2 CC1(C)C2CN(C(=O)C(c3cnn(C)c3)NC(c3cnccc3C#N)=O)CC12 S(=O)(=O)(CCC(=O)NCC(C)N(C(=O)COc1c(Cl)cccc1Cl)C)NC C1(OC)CCN(C(=NCc2cccs2)NCC2CCCN(CC(C)C)C2)C1 C#Cc1cnc(Nc2cc(O)ccn2)cc1C CC(C)=C=CC(=O)NCC1CC(C(N2CCC(O)(C(C)C)C2)=O)CO1 CN=C(NCC1CC12CC2(F)F)N1CCC(n2cccc2)CC1 N1(C(C(C(CC)C)N(C)C)=O)C(C(=O)NCC2CC2(F)F)CC2CCCC12 N1(C(c2c(C)nsc2)=O)C2CCC(C(N3CC(S(C)=O)C3)=O)C1CC2 CP(C)(=O)c1ccc(C(=O)NCC2(O)CCN(c3ncc4ccnc-4[nH]3)CC2)o1 N1(C(Cc2ccc(C(C)=O)s2)=O)CCCC(CNC(=O)Cc2ccn(C)n2)C1 C=CC(C)(C)CCNC(=O)CCC1CCC(NC(c2ccc(O)cc2)=O)C1 C12(C(=O)NCCCCC=C)CC(CN1C(c1sncc1C)=O)C2 C12CCC3(CC(C3)C(=O)N1)O2.C(CCCC(=O)OC(C)(C)C)N(C)C c1(C(N2C(CNC(CC3ON=C(CC)C3)=O)COCC2)=O)cccc2[nH]ncc12 c1(CCC(=O)NCC(C)(O)CNC(C2CC3(CCC3)C2)=O)nncnc1O C(=O)(C(C(C)(C)C)n1ccnn1)NC1CC(CNC(C=CCC)=O)CC1O c1(C(N2CC(CC)(NC(=O)CC(C)(C)OC)C2)=O)cc(C)nnc1O c1(C(N(c2cn(CC)nc2)C(c2c[nH]cc2C)=O)=O)cccc(O)c1 N1(C(CSCC#C)=O)CCC2(CCCN2C(c2cccc(P(C)(C)=O)c2)=O)C1 C=CCCCCC(C(=O)NCCCOC)N1CCC(O)(C(=O)OCC)CC1 C1(C(=O)NC(C)=O)CCOCC(=O)N1.N12CC(C1)C2=O.C(N)(=O)NC.O CC(C)CCCCCC(=O)N(C(C)CNC(C1CCC(F)(F)C1)=O)C C(C(F)(F)C(C)(C)O)NC(COCC(=O)N(c1ccccc1)C)=O c1(-c2cnc(OC)nc2)cnc2cc(C(=O)NCc3cc(F)cc(Cl)c3)[nH]c2c1 c1(CC(N2C3CN(C(CCC(C)OC)=O)C(C3)C2)=O)ncn2c1COCC2 N1(C(c2cnn(CCNC(C3(F)CCOC3)=O)c2)=O)CC2CC1CS2=O c1(C(=O)NCCC(C(=O)NC(CC#C)C(N)=O)OC)cc(O)ccc1C n1(CC(=O)NCCNC(c2c(C)oc(C#N)c2)=O)nc(C(F)(F)F)c2c1CCC2 N1(C(C(CNC(C2CCN(CC)C2)=O)C(C)C)=O)CC(C2=NOCC2)C1 CC1(C)CCC(C(=O)NC23CC(C(N4CCN(C5CC5)CC4)=O)(C2)C3)C1 N1(C(C(CO)NC(N)=O)=O)CCC(C2CC2)(NC(C2CCCSC2)=O)C1 c1(CCNC(=NCCC)NCC2(CF)CCC2)c[nH]c2cc(OCC)ccc12 C(C1=NOC2CCCC12)NC(C1N(C(c2cc(C)c(C)nc2)=O)CCC1(C)C)=O C1(C(N2CC(C)C(CNC(=O)CN3CC4CC4C3)C2)=O)COc2ccccc2O1 C1(CC(=O)NC(C)C)(C(=O)N(C)CC2CCN(C(c3ccon3)=O)C2)CCCC1 c1(C(=O)OC)cncc(OC(c2nc(OCc3ccccc3)sc2Cl)=O)c1 c1(-c2c(C(N(C(c3cn(CC4CCCC4)nn3)C)C)=O)nco2)ccc(Cl)cc1 Cc1ccc(C)c(OCCSc2ccc(C#N)cc2)c1 c1(CCC)nc(C)c(C(=O)NCC2(OC)CN(C(=O)CC3SC(=N)NC3=O)C2)s1 n1(CCCC)nc(C)c(C=CC(=O)NC2CCN(C(C3(C)CC3(C)C)=O)C2)c1Cl C1(C(=O)NC(CC)C(C)CN(C)C)CC2CCC1N2C(=O)C=CC1CC1 C1(C)(NC(CCC2C(C)C2)=O)CCN(C(=O)CN2CCCC2=O)C1.Cn1cnnc1 N1(C(=O)Nc2ccc(CCC)cn2)CCC(c2ccc(C)cc2)C1(C)C c1(C(N(C)CC2(CNC(C3C4CCN3CC4)=O)CC2)=O)cc2occc2n1C Cc1ccc(C(N2CCC(N(C(=O)CCc3cccn3C)C)C2)=O)cc1C c1(CC)cc(C(N2CSCC2C(=O)NC2(C(N)=O)CCOC2)=O)ccn1 N1(C(c2ccc(Cl)s2)=O)CC2CCC(C1)N2C(C1CCOCC12CCC2)=O c1(C(=O)NCC(=O)NC2(CNC(c3cccs3)=O)CCOC2)ccc(F)c(F)c1 C1(C(=O)NCCOCC2CCOC2)CC2CC1CC2NC(C1(C2CC2)CC1)=O C#CCC(CC(F)F)C(=O)NCC12CC1CN(C(=O)CC(O)CCCCC)C2 C1(NC(c2scc(C)c2C)=O)CCN(C(=O)CN2C(=O)CN(C)C2=O)CC1C CCC(C)(C)C(O)C(=O)N1CC(CNC(=O)CCc2ncc(C)[nH]2)C(O)C1 CC(C)CC(C)N(C)C(c1ccoc1CNC(c1coc(C2CC2)n1)=O)=O Cc1cc(CCCNC(=O)C2CC2)no1.C12CCCN1C(=O)CCCNC(=O)N2 c1(C(=O)NCC(C(C)C)NC(c2c(C)[nH]cc2)=O)oc2cc(Cl)ccc2c1C C1(NC(C2C(C)(C)CO2)=O)COCCN(C(=O)CCOC2CCOCC2)C1 C(=O)(CCCC(C)(C)C)N1CCC(C(C)C(N2CCCC2c2ccon2)=O)CC1 C1(CNC(C=C(C)C(C)C)=O)COCCN1C(=O)C(c1ccc(N(C)C)cc1)C N1(C(c2cc(C)oc2C)=O)CC(C)(C)CC1CC(N1CCCC(C(F)F)C1)=O c1(C(N2C(CO)CC(NC(CC3(N(C)C)CCCC3)=O)C2)=O)ccc([N+](=O)[O-])[nH]1 C(N=c1[nH]c(=NCc2cc(C)n(C)n2)[nH]c2c1CCCC2)c1cc(C)cc(Cl)c1 c1(CNC(C(=O)N(CCCC(=O)NC)C)=O)ccc(OC2CC2)nc1 n1(CC(=O)NCC(C)CNC(=O)Cc2csc(Cl)n2)cnc2sccc2c1=O n1(CC(=O)N(CCCNC(C(CCCC)(C)F)=O)CC)c(C)cc2ccccc12 C(=O)(C1Cc2ccc(F)cc21)N1CC(COC)N(C(c2ncncc2Cl)=O)CC1 C1(C(=O)OC2CC(OCc3ccccc3)C2)CN(CC)CC1(C)C c1(CC)nonc1C(=O)NC1CC(O)(CNC(C2CCCN2C(C)=O)=O)C1 c1(N2CCC(CCN(C(=O)C(O)CC3CCCCC3)CO)C2)ncnc2sccc12 C(=O)(C(CC(C)C)OC)N(CCCCCCNC(C1C(C(=O)OCC)C1)=O)C N1(C(=O)OCC=C)CCC(CC(=O)NC2CCC2NC(=O)COC(C)(C)C)CC1 C1(NC(c2cn(C(C)C)nn2)=O)CCOC(C(=O)NCCCc2cc[nH]n2)C1 N1(CCN(C(C(N2C(CC)CCC2)=O)=O)C)CCN(C(=O)COC)CC1 N1(C(=O)C(F)=C2CC2)CCCC(N(C(=O)Cc2c[nH]ccc2=O)CCO)C1 c1(C(=O)NCCCN(C(CCC(C)C)=O)C(C)C)cccc2ncsc12 c1(C(=O)NC(CNC(C(C(C)(C)C)OC)=O)C2CCC2)ccc2oc(S)nc2c1 CC(CC(C)(C)C)C(=O)N(CCCCNC(=O)CSCC(N1CCCCC1)=O)C C1(NC(C2(C3N(C(CCC=CC)=O)CCC3)CC2)=O)CCCC(n2cccn2)C1 N1(C(CC(C)F)=O)CCC(O)C(NC(=O)C(C)NC(=O)C2CC2)C1 C1(C(=O)NC2CN(C(CC(CC)C)=O)CC2SC)CCn2cncc2C1 N1(C(C(CCC2CCC2)NC(CC(COC)(C)C)=O)=O)C2CCC1CC(=O)NC2 CN1CCCCC(C(=O)NCC2CC(O)(CNC(=O)CC(F)(F)Cl)C2)C1=O C12CCCC1NC(=O)C2.C1(N(C)C)CC(C)(NC(=O)CC2CC3CC3C2)C1 C(=O)(C1=NNC(=O)C1)NC1(CC=C)CN(C(=O)COCC2CCCO2)C1 N1(C(C2(C)CC(=C)C2)=O)CCN(C(C2CC(OC)C2)=O)C(c2nccn2C)C1 Cc1nc(=NC(C)CN(C)C(c2cc(F)c(F)cc2F)=O)s[nH]1 C(C)(CCCCO)NC(CC1CC(NC(C(CC)=CC)=O)C1)=O CC(C)(CCCO)C(=O)N1CCCC1C1CCN(C(=O)Cc2csc(Cl)c2)C1 C1(CNC(c2cn(CC=C)nn2)=O)CC(C)(C)CN1C(c1csnc1Cl)=O c1(C(=O)OC)c(N2CC(C(N)=O)(CNC(=O)C(C)(F)F)C2)ncnc1Cl Cn1cc(CCSc2ccccc2)c(NC(=O)NCCCc2ccc(O)nc2)n1 C1(C#N)(C(=O)NCC(CNC(c2cnc(C(C)(C)CF)o2)=O)OC)CC2CC2C1 N1C(=NCCNS(=O)(=O)NC)NCC2(C1CCC(C)C)CC2 N1(c2nc(C)cc(OC)n2)CC2(C1)SCCC2NC(=O)Cc1ccccc1C C1(CC(=O)NCCCCC(=O)OC)C2CCC(C2)N1C(C1CCC1C)=O Cc1nc(Cl)nc(N(C2CCCN(C(c3cc(Cl)c(Cl)n3C)=O)C2)C)c1F C(=O)(CC(C)(C(F)(F)F)N(C)C)NCC1N(C(=O)OC(C)(C)C)CCC(O)C1 Cc1occc1CC(=O)NCC1CC1CNC(C1(Cc2cccnc2)CC1)=O N1(C(CC=C=C)=O)CC(NC(c2nccnc2-n2ccnc2)=O)CC12CCOC2 C1(C(=O)N)CC2(CC2)CN1C(c1cnc(CO)s1)=O.C1(N2CCCC2)(C)CCC1 Cn1cc(S(=O)(=O)NCC(=O)NCC(C)(C)CNC(C2(C)CC(C#N)C2)=O)cn1 C(=O)(C1=CCCC1(C)C)N(C)CC1CCN(C(C2C(C)(C(C)C)C2)=O)CC1 c1(NC(C2CC3CC3N2C(c2ccc(Br)cc2O)=O)=O)ccc([N+](=O)[O-])c(Cl)c1 c1(C(=O)NC(C2OCCN(C(C)=O)C2)C)cc(Br)cnc1O CC1CCN(C(C2CCC(=O)N2C)=O)CC1NC(c1cn(CCC2CC2)nn1)=O c1(C(N(C(CC)CNC(=O)C(C)OC)C)=O)cc(OC)cc(F)c1 C1(OCC(C)C)CCCN(c2nnc(C3CCC(=O)N3)n2CC2(C)CCCC2)C1 c1(C(=O)NCC(C)CN(C)C(c2coc(Cl)n2)=O)cc2ncccc2[nH]1 c1(NC(Cc2ccc(-c3cnc(C(=O)OC)s3)cn2)=O)ccc(Cl)cc1F C1(C(=O)NCC(CCNC(=O)C(C)=CC(C)(C)C)OC)CCc2nnc(O)n2C1 c1(C(=O)NCC(CO)NC(c2cnc(CC)[nH]2)=O)ncncc1OC C(=O)(C(C)C(O)C(C)CC)N(C(CC)CC(N1CC2CC1CS2=O)=O)C c1(OC)cccc(CC(=O)NCC(O)CNC(c2c(C)csc2C)=O)c1 c1(C(=O)NCC2C(C)CCN(C(=O)C=Cc3cn[nH]c3)C2)nc2ccccn2n1 c1(C(C(=O)NCCCCCC)N(C)C)c(C)nn(Cc2ccc(F)cc2)c1Cl C12(NC(c3c(C)cncc3C)=O)CCCC1N(C(c1ccc(Cl)cn1)=O)CCC2 C1(NC(C2(C#C)CC2)=O)CC12CCN(C(=O)CCCC1CCCO1)C2 N1(C(C(C)c2ncco2)=O)CC=C(c2cccc(F)c2F)CC1 Cc1c(NC(c2ccnc(-c3ccoc3)c2)=O)cnn1-c1ccc(F)cc1 CCC(C)(C(=O)N(C)CCN(C(=O)CSCc1cccc(C)c1)C(C)C)OC C(=O)(CC1=CCOCC1)N(C)CC.C(=O)(CCC(=O)c1cnn(C)c1)NC1CC1 c1(CCC)ccc(OC(C)C)c(C(C(=O)NCC2CC2)N(CCOC)C2CC2)c1 c1(C(N(C2CCN(C(c3cn(CC)nc3)=O)CC2C)C)=O)scc2c1CCCC2 Cc1noc2cc(C(N3CCC(C(F)CNC(=O)CCF)CC3)=O)ccc12 N1(C(C(C)CC(F)(F)F)=O)CCCCC12CN(C(=O)CN1CC=CC1)C2 c1(C(=O)NC2CC(F)CN(C(c3ccncc3)=O)C2)ccnn2ccnc12 C(CCC(=O)N1CCCC1C(=O)NCC1CC1)OCC=C c1(C(=O)OC)cccc(C(=O)NCCOC2CCN(C(C3CCSC3)=O)C2)c1O C(=O)(C(F)(F)C(F)(F)F)N1CC(N(C(=O)C(O)C2CCC2)C)C1 C1(C(=O)NC2CC(NC(CC(C)(C)F)=O)C2)COc2cc(F)ccc2C1 c1(C(C(=O)N(C)CC2CCCC2)NC(C(C)n2ccnc2)=O)cn(C)nn1 N1CC(CO)C(C)(C)C1.C(C)(CC(C)(C)C#N)c1cn(C(COCC)C=O)nn1 C1(C2CCOCC2)(C(=O)NCC=CCNC(=O)C(c2ccccc2F)O)CC1 c1(NC(C2C3C(NC(CC4C(=O)NCC4)=O)C4C(C3)C42)=O)ccc2nccn2c1 Cc1cc(O)nnc1C(=O)NC1CCN(C(c2cc(F)c[nH]2)=O)C(C)C1 Cc1ncc2n1CCC(C(=O)NCC13CC(CN1C(=O)Cc1cscn1)C3)C2 C1(NC(C(CCC#C)NC(c2cn(C)c(C)n2)=O)=O)C(=O)OC2CCCC12 C=CCC(CNC(=O)C(C)NC(=O)COC)NC(=O)Cc1cc(COC)no1 c1(CC)cc(C(=O)NC2CC(CNC(=O)C(C#N)CC)C2)cc(Cl)c1 C1(C(=O)NCc2ccc(O)c(F)c2)CC12CCN(C(=O)CCC(F)(F)F)CC2 c1(N2CCC(CNC(=O)NCCCSC)C2)ccc(F)cc1F C(c1ccncc1)=C(C)C(=O)NC(C)(C)CNC(=O)C(c1ccc(Br)s1)C c1(C(N(C)CC2(CC(C)C)CC2)=O)cc(CNC(=O)COC(C)(C)C)ccn1 N1(C(c2c(OC(C)C)nccc2)=O)CC2CCC1(CNC(=O)C1CC1)CC2 N1(C(Cc2nc(C)oc2)=O)CCN(C(=O)C(C)(C)C(C)O)CC1C(C)C C1(C(=O)NCC2(C)CC(C)(C)C2)N(C(=O)Cc2ccc[nH]2)CCCC1(C)C C(=O)(C#CC1CCOC1)NCCCCCN(C(=O)COCCNCC(F)(F)F)C c1(C(N2CC3C(NC(=O)CN4CCCC4)C3C2)=O)cc(Cl)ccc1Br N1(C(C2C(C)C2)=O)CCC2CN(C(=O)CC(C)CNC(=O)OC(C)(C)C)CC12 N1(C(C)CC(=O)NCCCCCN(C(=O)CC2CCCC2O)C)CCCCC1=O C=C1CCC(C(=O)N(C(CNC(c2c(C)nsc2NC2CC2)=O)C2CC2)C)CC1 C#Cc1ccc(C(N2CCC(C)CC2C(N2CCC(COC)CC2)=O)=O)c(C)c1 C1(F)(CNC(c2nc(CC(C)C)sc2)=O)CCN(C(=O)C=CC(C)(C)C)C1 C1(c2n(CCOC)nc(-c3cccc(C)c3)n2)CCn2c(nn(C)c2=O)C1 Cn1nc(C(=O)NCCNC(C2C(c3ccccc3)C2(C)C)=O)c(Br)n1 C1(NC(Cc2c(C)ccs2)=O)CC2CCC(C1)N2C(=O)CCCc1cccnc1 C=CCC(CC(C)C)C(=O)NC(C(N1CCOC(C=C)C1)=O)C1CC1 CCCC(CC)CC(=O)N(CCCNC(c1cc2scc(C)c2[nH]1)=O)C(C)C c1(C(=O)OCc2ncn(-c3ccccc3)n2)ccc(F)c2cccnc12 C1(Nc2ncc(C)cn2)CCCC12CN(C(c1ccc(C)c(O)n1)=O)C2 Cc1cc(C(N2CC(N(C(=O)Cc3ccco3)C)C(F)C2)=O)c(O)c(C)c1 N1(C(Cc2nc(C)sc2)=O)CCC(NC(C2C(C)(C)OC2(C)C)=O)CC1C N1(C(c2n(C)nc(Br)c2)=O)CC2CN(C(=O)CCc3ccccc3O)CCC12 c1(CO)ccsc1C(=O)NC1CC(C(F)F)C1.C12(CCC1)CC(=O)NCC2 c1(C(N2CC(NC(Cc3ccc(OC)cc3)=O)C(C)(C)C2)=O)cc(C)c(F)c(C)c1 c1(C(N(CC(C)CNC(=O)C(C)(F)F)C)=O)c[nH]c2cc(Br)ccc12 Cc1ccc2[nH]c(C(N3CC(CNc4ccc([N+](=O)[O-])cn4)C(C)C3)=O)cc2c1 Cc1cc2c(o1)CC(C)(C)CC2NC(=O)N=c1ccn(-c2cncnc2)[nH]1 c1(C(N(CC(CC)NC(=O)CCC2CCC(=O)N2)C)=O)cc(C)n(C(C)(C)C)n1 N1(C(C)C(=O)Nc2cccc(F)c2)CCCCC(N2CCN(C)CC2)C1 C(=O)(C1=CC2CCCCCC12)N1CCC(NC(C2(NC(C)=O)CCCC2)=O)C1 C1(C(=O)NCC(CC)Nc2ncnc(O)c2Br)CCc2nc(C)ncc2C1 N1(C(CN(C(=O)OCC)C)=O)CC2CC2(NC(=O)Cc2cc(CC)no2)C1 C(C)(C(=O)N(C)CCN(C(C1(C)CC1Br)=O)C(C)C)OCCOC c1(N2CC(C)OCCC2)nc(NC2COCCOC2)c2ccsc2n1 c1(C(=O)NC2C(NC(c3c(OC)n(C)nc3C)=O)C2)cc(Cl)ccc1[N+](=O)[O-] c1(C(=O)Nc2nnc(NC3CC4COCC4C3)s2)cc2ccccn2n1 CC1=NC(C(=O)N(C)CC2CN(C(=O)CC(C)c3cnn(C)c3)C2)CS1 C1(NC(c2c(C)n[nH]c2C)=O)CCCCN(C(=O)CCc2ccccc2F)C1 Cc1ncccc1CCC(=O)NCC(c1ccccc1)NC(=O)Cn1cnnc1 Cc1ccc(CC(=O)NC2CCCC2CC(N2CCCC(C(C)(C)C)C2)=O)cc1 c1(CCC)ncc(C(N2CCCC2CCNC(=O)CCNC(=O)CO)=O)s1 c1(C(=O)NCC(C)(C)NC(C2C(COC)C2)=O)c(C)nn2ncccc12 C1(CNC(C(CC)NC(=O)CC2(N(C)C)CC2)=O)CCCOC1(C)C C1(NC(C2(COC)CCC2)=O)CC(C(N2CCCC(NC)C2)=O)CC1O C1(NC(CSCC(N)=O)=O)CC2CCC1(CNC(c1nn[nH]c1Cl)=O)C2 CC1(C)CCC2(CC1)CC2CNc1cncc2nccn12 C1(NC(c2n(C(CC)(C)C)nnn2)c2ccc(SC)o2)(OC)COCC1CS(C)(=O)=O CC1(C)CC(C)(CNC(C2(C)CC2(F)F)=O)CN1C(=O)CN1CC=CC1 c1(C(N2CCC(Cc3ccccc3)C2)C)nc2c(s1)CCC2 c1(C(=O)NC(CNC(C2C(OCC)C2C)=O)C(C)(C)C)cc(C)n(C)c1C C1(N(C)C(c2ccn(C)n2)=O)CCCC2CN(C(C34CCCC3C4(F)F)=O)CC12 c1(OCC(=O)OC(C(CC)OC2CCCC(C)C2)=O)cccc2ccccc12 c1(C(CC)C(N2CCN(C(C3CC3F)=O)C(C)C2)=O)cccc2ccccc12 N1(CC)CC2CN(C(C3C=CCN3C(=O)C(c3cncnc3)C)=O)CC2C1 C(=O)(C(F)C(=O)NCc1n[nH]cc1C(=O)NCC(C1CCOC1)O)OCC Cc1cc(C)nc(N2CCCC2C2CCN(C(=O)C(O)C(C)C)C2)n1 C1(NC(C2C(CC)OCC2)=O)CN(C(=O)CCC(C)SC)C2CCCCC12 N1(C(c2cc(C(=O)OC)ncc2)=O)CC2(CCN(C(C3CC=CCO3)=O)C2)C1 C1(N(C)C(C2CCCSC2)=O)CCC2CN(C(=O)C#CC(C)(C)O)CC12 C=CC(O)C(=O)N(CC(CC)NC(C1CCCN1C(=O)C1CC1)=O)CC N1(C(CC(CC)OC)=O)CCC(CCNC(C2(Cl)CCC2)=O)CC1C c1(CN(C=O)CC(c2ccc(Cl)c(Cl)c2)O)cc(Cl)ncc1Br CC(CO)(C(F)(F)F)NC(C1CN(C(C23CC(C2)C3)=O)C1)=O S(=O)(=O)(c1cc(C(=O)NC(C)C(C)NC(c2ccc(=N)[nH]n2)=O)co1)NC C(=O)(C(C)(O)C(F)(F)F)N1C(C(=O)NCC(C)(C)C)CC(F)C1 c1(N(c2nnc(C3(C#C)CCCC3)n2CC2CCCCO2)C)cnc(Cl)cc1C N1(C(C(=O)NCC2(N3CCCC3)CCC2)=O)CCC(O)(Cc2ccc(F)cc2)CC1 Cc1cc(O)ncc1CNC(C1CC=CCN1C(=O)C=CC(C)(C)C)=O C1(NC(c2c(C)cnnc2)=O)CCSC12CN(C(=O)C(N1CCCCC1=O)C)C2 c1(C(=O)NC2CCC2NC(C2C3CCCCC23)=O)c(Cl)ccc2cccnc12 c1(OC)ccc(C2CCCN2C2CCN(C(=O)OC(C)(C)C)C2)cc1 c1(C(=O)NC(CCOC)CNC(c2cnc(-c3cccs3)o2)=O)c(Cl)cnn1C c1(CC(=O)NC2C(C)CN(C(=O)C=CC3CCCN3C)C2)cnc2cccnn12 S(=O)(=O)(C1CN(C(C2CCCOC2)=O)C1)N1CCN(C(c2c(C)ocn2)=O)CC1 C1(C(N2CC(NC(CC3CC(=C)C3)=O)C(C)(C)C2)=O)CCCCN(C)C1=O N1(C(c2c(CC)ncs2)=O)CCCC(C2(NC(=O)CC(F)(F)F)CC2)C1 c1(C(=O)NC2CCCC(CNC(C(C)(C)N(C)C)=O)C2)cc2c[nH]nc2s1 C1(NC(C2CCC(C)N2C(c2ncccc2Cl)=O)=O)CC2CCCCC12 Cn1nnc(C(=O)NCC2OCCC2C(N2CCC(C(C)(C)O)C2)=O)n1 c1(N2C(CNC(=O)CC3CC(F)C3)CCCC2)ccc([N+](=O)[O-])c(O)n1 CCCCC(CN=c1[nH]c2cc(Cl)ccc2s1)NC(=O)CCC1CCC(=O)NC1 C1(CC(=O)N(C(c2cc(C)on2)C)C)(NC(C2CCC(C)(C)C2)=O)CCCCC1 N1(CCC(=O)N(c2ccc3c(c2)OCO3)C(C)=O)CCCC2(C1)CC2(F)F N1(C(CC(C)N(C(C(CC)SC)=O)C)=O)CC(O)C2(CCCC2)C1 c1(SCC)cccc(CC(=O)NC2CCN(C(=O)C(CO)NC(N)=O)C2)c1 N1(C(=O)N(Cc2ccns2)CC2CC2)CCC(C(N2CCOCC2)=O)CC1 C1(C(N(C(C)C)CCN(C)CCO)=O)CC1C N1(C(CC(CC)C(F)F)=O)CCCC(C2CN(C(C3(C)CC4(CCC4)C3)=O)C2)C1 N1(C(C(=O)NCC=C)c2nc[nH]n2)CCC(Oc2ccccc2)C1 c1(CN(C(=O)NC2CCCC2)CC)cc(OC2CN(CC)C2)ccn1 C=C(C)C(O)CC(=O)N(C1CN(C(C2CCC(=C3CCC3)CC2)=O)C1)C C1(C(C)C(=O)NC2(CC3CC3)CC2)CCCN(C(c2cc(=N)[nH][nH]2)=O)C1 C1(N(C(C(C)OCC#C)=O)C)CCCCC1NC(c1cc(C(C)C)oc1C)=O CCC(C)(CNC(C1CN(C(c2ccc(Cl)o2)=O)CCN1C)=O)C(N)=O c1(C(=O)NCC(CNC(CSCCCC)=O)C)cnccc1C Cc1cc(C(=O)NC(C2CCCCC2)CNC(=O)COc2cnn(C)c2)oc1C N1(C(c2nc(C)c(Br)s2)C(=O)NCCCSC)CC2CCC(C1)C2(F)F c1(NC(C2(C)CNC(=O)C2)=O)ccc2nccn2c1 CCC(CC(=O)N(CCNC(C1CN(C(C)C)C1)=O)C1CC1)OC N1(C(C2(C(=O)OC)CC2)=O)CC(C(F)(F)F)CC1CO CC(C(CO)NC(=O)Cc1csc(C(F)(F)F)n1)NC(C1COC(=O)N1)=O C1(NC(CCN(CC(F)(F)F)C)=O)C2CC1N(C(C1CCCCO1)=O)C2 C1(S(C)(=O)=O)(C(=O)NCC(C)(C)NC(=O)Cn2cnc(C#N)n2)CCCCC1 N1(C(COCCCC)=O)CCC(CNC(c2c[nH]nc2OC)=O)C1(C)C C1(C)(C(=O)NC2CC3CN(C(C4CCC(C)CC4)=O)CC32)CCC(F)(F)CC1 c1(CN2CC(C(=O)NCC3CC4C=CC3C4)C(O)CC2)c(O)ccc(F)c1Br c1(C(=O)NCCCCN(C)C(C2CCC2CF)=O)cnc(C2CC2)o1 c1(NC(C2(CC)CC2)=O)ccccc1NC(C1CCCCN1C(=O)OC(C)(C)C)=O c1(C(N2CCC(CNC(C3CC(C)(C(=O)OC)C3)=O)C2)=O)ncccc1C C12(C(=O)NC3C(OC)C(O)C3)CCC(CN(C(=O)C(F)C(C)(F)F)C1)C2 c1(C(=O)NCC(CCCC)NC(=O)C(CCC)N(C)C)ccc(N)cc1[N+](=O)[O-] C#Cc1cnc(=NCC(C)N(C)C(c2cnccc2C)=O)[nH]c1 C(N=c1cc(NCc2cccnc2N(C)C)nc[nH]1)c1cn(CCN(C)C)nn1 C1(NC(CCc2ccc(OC)nc2)=O)CN(C(=O)Cc2ccsn2)C2(CCC2)C1 C(=O)(C(C(C)OC)OC)N1C(C)(C(=O)OC)CC1.C12CCC(CC1)NC2=O C1(NC(c2csc(Cl)c2)=O)C2CN(C(=O)C(Cc3ccccc3)C3CC3)CC12 c1(CCC)cc(C(=O)NC2COCC2NC(C2(OCC)CCOC2)=O)cc(O)n1 N1(C(c2cc(C)ns2)=O)CCCC(O)(c2cn(CC3CC(F)(F)CO3)nn2)CC1 C(CC(CNC(C1(Cl)CC1(F)F)=O)OC)NC(CCN(C(CCC)C)C)=O n1(C(CC)C)ncc(C(=O)NCC2CCN2CC(c2ccccc2)O)c1C1CC1 O=C1CCC(CC(=O)NCc2ccnc(C(=O)NCC3CCC3)c2)CN1 N1(C(c2c(C)noc2Cl)=O)C2CCC1CC(NC(=O)C(C)(O)c1ccccc1)C2 c1(NC(C(CN(C)C)NC(CC(C=C)(C)C)=O)=O)c(C)ccn(C)c1=O c1(C(=O)NC2C=CC(CNC(C3(C(C)(F)F)CC3)=O)C2)ccc(F)c(C(F)F)c1 C(=O)(CCCCCCBr)N1CCN(Cc2cccc(C)c2I)C2C1C2 C1(NC(C(=O)O)Cc2ccc(F)c(Cl)c2)CCC2(CCCCC2)C1 c1(C(=O)NCC2C(NC(C=C(C)C(C)(C)C)=O)C2)ccc(C(C)C)nc1C(C)C N1(C(C=CSC)=O)CCN(C(C2CCC2C(F)F)=O)C(c2ccc(CC)cc2)C1 c1(CC)cnc(C(=O)NCC2CCCCN2C(C2(C)CCCO2)=O)nc1 C1(=CC(=O)NC(C2CN(C(c3ccc(O)nc3)=O)C2)C)C2CC3CC(C2)CC1C3 N1(C(C2(C(C)C)CC2)=O)C2CCC1(CNC(=O)CCc1ccc(O)nc1)CC2 C1(F)(CNC(C(c2ccnn2C)C)=O)CCCN(C(C2(C)CCOCC2)=O)CC1 Cc1ccc(O)cc1CCCC(=O)NCC1CCN1C(=O)C(C)(F)F Cc1n[nH]cc1C=CC(=O)NCC1CCN(C(=O)C(C)NC(=O)C2CC2)C1 c1(OC)ccc2c(c1)OCCC2NC(c1ccc2sc(C(F)F)nc2c1)=O CC1CC(C(=O)N2CCC(C(C)(C)NC(c3cnc(N)cn3)=O)C2)=NO1 C1(C(C(=O)N(CC=C)CC2CC2)C)CCCN(C(=O)CC2C(C)(C)C2(C)C)C1 c1(C2(C(=O)NCC(CN(C(CCOCC#C)=O)C)O)CC2)ccc([N+](=O)[O-])cc1 Cc1ccccc1C(C)C(N1CCOC(CNC(=O)CC2CC2C)C1)=O N1(C(Cc2c(Cl)cn(C)n2)=O)CC2CCOC2(CNC(C2CCCCO2)=O)C1 c1(C(N2CC3CC3(C(C)C)C2)C(=O)NCCCOC)ccc(C2CC2)cn1 N1(C(c2c(C)n(C(C)C)cc2)=O)C2CCC1CN(C(c1ccnc(F)c1)=O)CC2 c1(C(=O)NC(CNC(C2CCC(CCC)CC2)=O)C)c(C)nn(C)c1Cl N1(C(N)=O)CCC(C(=O)NCCOCCOCCNC23CCCCC2C3)CC1 c1(CNC(C(c2cnn(C)c2Br)N2C(CC)CCC2)=O)cc(C2CC2)ccc1F C(=O)(C1=NOC2(CCC2)C1)N1C(CC(=O)NCC(O)C2(Cl)CC2)CC2(CC2)C1 C1(NC(CC2CC(C)N(C(C3CN(C(N)=O)C3)=O)C2)=O)C(O)C2CCOC12 C(=O)(CC(CC)N(C(=O)C(C)CC#N)C)NCc1n(CCC)cnc1 C1(C(C)C)CN(C(c2cnn(C)n2)=O)CCN1C(c1ncc(Br)cc1N)=O CN1CC(C(N2CCC(N(CCO)C(=O)Nc3cnccn3)CC2)=O)CC1=O c1(C(=O)NCC2(F)CC(NC(C3CCC(=O)O3)=O)C2)ccncc1C(F)F CC1CN(C(c2sc(N(C)C)nc2Cl)=O)CCC1CNC(=O)C(C)(C)C#N Nc1ccc(CNC2CCC(C(=O)NCCOC(F)(F)F)C2)cc1[N+](=O)[O-] c1(C(=O)NCCN(CC(C)O)C(=O)CC2CC3CC3C2)ncc(Br)cc1N Cc1nnc(O)c(C(=O)NCC2C=CCN2C(=O)C(c2ccc(Cl)s2)=O)c1C C1(C(N2C(CN(C(C(CC3CCCC3)OC)=O)C)CCC2)=O)COC(=O)N1C C(=O)(C1CSc2ccccc21)N(CCC)CCNC(c1cnc(C(F)F)nc1)=O c1(C(=O)NC2Cc3ccc(Cl)cc3C2)ccc2[nH]c3ccccc3c2c1 Cc1nc2ccc(C(=O)NC(C)C(C)NC(=O)CCC(C)(C)F)cc2n(C)c1=O C(=O)(C(CC(C)C)C(C)C)NCC1(CNC(c2c(Br)ccc(C)n2)=O)CC1 C1(C(=O)NCC2(CNC(C3(C)CCCCC3)=O)CCC2)CCn2nnnc2C1 N1(C(C(C=C)OC)=O)CC2(CCN2C(=O)C(N2CCSCC2)C)C1 C(=O)(C#CC1CCCO1)NC1CC(F)(CNC(Cc2n[nH]c(=N)s2)=O)C1 C12(CNC(c3c(CC)noc3)=O)CCC(CC1NC(=O)C(=O)NCCC(N)=O)C2 NS(=O)(=O)c1cc(Cl)c(NCC2CC3(CO2)CC(F)(F)C3)c(Cl)c1 c1(C(=O)NC2CCN(C(C3CN(C)C(=O)C3)=O)C3C2C3)cc2c(nc1O)CCC2 N1(C(c2cc(C)ncc2)=O)CC(C)CN(C(c2cc(O)cc(O)n2)=O)CC1C N1(C(C2N(S(C)(=O)=O)CCCC2)=O)CC(CNC(=O)Cn2cccc2)C2(CC2)C1 C(=O)(C(C)S(N)(=O)=O)N1CCCC(CN(C(C2N(CC)CC2)=O)C)C1 N1(CC)OCC(NC(C2CC(O)CN2C(=O)CCOCC(C)(C)C)=O)C1=O CCC(O)C(C)C(=O)N(CCCNC(c1c[nH]nc1-c1cccc(Cl)c1Cl)=O)C C1(N(C(c2ncc(C)nc2)=O)C)CCN(C(C2CC2C(C)(F)F)=O)CC12CC2 C(CC(C)(C)C(=O)NC1CCCC(NC(c2cnc(O)s2)=O)CC1)OC c1(C(=O)NCC2(F)CN(C(CC(C(F)(F)F)OC)=O)C2)ncc2c(F)cccn12 c1(CC)cc(C(=O)N(C)CC2CCCN2C(c2cscc2C(F)F)=O)c(C)o1 C(CCCC(C)C)(C(=O)NCCCOC)N(CC)Cc1cccc(Cl)c1C c1(CNC(c2cnc(CNC(=O)OC(C)(C)C)o2)=O)ccnc(Cl)c1F C1(C(N2CCC(C(=O)NCCC3CC3CCCO)(CC)C2)=O)CC(=O)NC(=O)C1 C=C(Cl)CC(C(=O)NCc1cnn(C)c1C)NC(=O)C(C)COC(C)=O C(=O)N=c1[nH][nH]c2ncc(Br)cc12.Cc1ccc(C2CC2)s1 N1(C(CCOC(C)C)=O)CCC2CCN(C(c3ccc(C4CC4)cc3)=O)CC2C1 C(=O)(C(C)CC(F)(F)F)NC1(C(=O)NCC#C)CC(F)(F)C1 C1(CN(CC(=O)N(CCC)CCC)C)CCN(C(=O)CC2(O)CCOC2)C1 Cn1nccc1C(O)C(=O)NCCC1CC(NC(=O)COCC2(F)CC2)C1 C1(C(=O)NCc2cc[nH]c2C(=O)NOC2CCOC2)(CC)CCCO1 O=NN1CCCCC1C(N1CC(F)(F)CC1CCNC(c1ccns1)=O)=O C=C(C)C1OCCC1C(=O)NCC1(CNC(C2(C(C)(C)O)CCC2)=O)CCC1 c1(CC(=O)NC2CC3CC2N(C(=O)CC2CC4CC4C2)C3)cnn2ccccc12 CC1CN(C(=O)CC2CCC3CC23)CCN(C(c2coc(C(F)F)n2)=O)C1 N1(C(c2cccc(Cl)c2O)=O)CC2CCN(C(c3ncoc3C3CC3)=O)C2C1 c1(C(=O)NCCN(C(=O)C2=CCCOCC2)C)cc2n(n1)CC(C)(C)CO2 C(=O)(CC1=CCN(C(c2ccc([N+](=O)[O-])o2)=O)CC1)NC(c1c(C)ncs1)C N1(CC(=O)N(C2CCN(C(C3(C)CC4(CCC4)C3)=O)C2)CC)OC(C)(C)CC1=O S(=O)(=O)(c1c[nH]c(C(N2CCC(NC(c3ncoc3C)=O)C2)=O)c1)NC C1(C(=O)NCCN(C(C2CCCN2N=O)=O)CC)CCN(C2CC2)CC1 Cc1ccc(=O)n(CC(=O)NC2CN(C(=O)C(c3cncnc3)C)CC2(C)C)n1 Cc1nc(CNC23CC(C(=O)Nc4[nH]cnc4C)(C2)C3)co1 N1(C(c2c(CC)cco2)=O)CCN(C(c2cn(C)cc2C)=O)C2CCCC12 Cc1c(Cl)ccc(C(=O)N(CCCCCCNC(=O)COCCF)C)c1Cl C1(NC(C2(C)CC2)=O)CCN(C(c2cnc(C3CC3)s2)=O)CC1O C(=O)(C(F)CC(CC)CC)NC1CCN(C(CC(C(=C)C)OCC)=O)CC1CO N1(C(C2C(=C)C2)=O)CC(NC(C2CCC(C(F)(F)F)CC2)=O)C(O)C1 C1(OC)(CNC(=O)CN2CC3CC3C2)CCN(C(=O)CC2CC(OC)C2)CC1 Cn1cnc(C(O)CNC(=O)CCOCCNC(=O)CN=[N+]=[N-])c1 c1(NC(CCCC=C)c2nnnn2CCCSC)cnc2ncccc2c1 N1(C(c2ccc(CCC)s2)=O)CC(OC)C(NC(c2nocc2C(C)C)=O)C1 CC1CCCn2cc(-c3nc(-c4cscn4)nn3CC3(C)CCCC3)nc21 Cc1c(C(=O)NCCCNC(c2occc2C2CC2)=O)cnn1C(C)(C)C N1(C(C(C)C(C)O)=O)CCN(C(C2OCCC2c2cnn(C)c2)=O)C2(CCC2)C1 C1(C2CCN(C(=O)C(c3cnccn3)C)C2)(NC(C2CCC(C)C2)=O)CC1 CCC(C(=O)NC1CCCCC1C(=O)NC1CC2(CCCCO2)C1)C(C)(C)CC Cc1cc(N2CCC(NC(=O)C(C)Cc3cnn(C)c3)CC2)nc(CCOC)n1 CC(CC(F)F)C(=O)NCC(C)(Cn1cccn1)NC(=O)CC1(O)CCOC1 c1(C(=O)NCC23CC2CN(C(c2cnoc2)=O)C3)nnc(O)nc1O c1(CNC(CN(C2CCSC2)C)=O)c(F)cccc1F C1(C(N(C(C2CCOCC2)C)C)=O)CCC(C)(C)N(C(=O)C(O)CCN(C)C)C1 c1(CCC(N2CCC(NC(COCCC=C)=O)C2C)=O)c(C)nc(O)nc1O N1(CCN(C(=O)CN2CCCC2=O)C)CCN(C(=O)CCCF)CC1 C1(NC(CCC2N(C)CCCC2)=O)CCSC12CN(C(C1CC1(F)F)=O)C2 C1(C(C)C)CN(C(=O)COCc2ccncc2)CCCN1C(=O)CCN(C)C C1(C2(O)CCC2)(CNC(C(c2cccnc2)NC(CC2CC(=C)C2)=O)=O)CC1 c1(CC)ccc(C(=O)N(C)CC2CN(C(=O)C(C)S(C)(=O)=O)CC23CC3)cc1N C1(c2cn(C3(C(=O)NC4(C)CSCO4)CC3)nn2)CC2(CC(OC(C)(C)C)C2)C1 C1(NC(C2CC3(C2)CC2(CC2)C3)=O)CC2COCC(C1)N2C(C1CC1Cl)=O C1(F)(CNC(CNC(C2C(C)C2)=O)=O)CC(CNC(=O)CN(C2CCSC2)C)C1 C1(N(C(COCCC=C)=O)C)CCC(NC(=O)CC2(C(F)(F)F)CCC2)C1 N#Cc1nc(=NCC(C2CCCC2)NC(=O)C2CCCn3cnnc32)c(Cl)c[nH]1 c1(C(=O)NCC2N(C(C(CC)F)=O)CCCC2C)ccncc1[N+](=O)[O-] c1(C(N(CCNC(c2ncc(C)c(C#N)c2)=O)C)=O)ccc(N=S(C)(C)=O)s1 c1(C(=O)NC2(COC)CN(C(C3CC3Br)=O)C2)ccc(F)cn1 c1(CNC2(Cn3c(C(N4CCC(O)(CO)C4)=O)ccc3)CC2)cc([N+](=O)[O-])n[nH]1 N1(C(C2(OC)CCCSC2)=O)CCC(O)C(NC(=O)CC2NC(=O)NC2=O)C1 CCC(C(=O)N1CCC(CC(=O)NCc2nc(OC)[nH]n2)C1)n1cccn1 N1(C(c2c(OC)c[nH]n2)=O)CC(NC(C2CC(n3cccn3)C2)=O)C(C(F)F)C1 Cc1ccc2oc(=O)c3cnn(CC(=O)NCC(O)CCNC(=O)CC#N)c3c2c1 C1(CNC(c2ccnc(F)c2)=O)CC(F)(F)CN1C(=O)C=Cc1ccsc1 c1(OCC=C)cccnc1C=CC(c1c(C(=O)OC)nn(C)c1Cl)=O N#Cc1cncc(CN2C(C(=O)NCCF)CC3CC23)c1 c1(CC(=O)NCC(CCNC(c2ccn(C)n2)=O)O)ccccc1S(C)(=O)=O C1(CNC(C(C=C)O)=O)CC2COCC2N1C(=O)Cn1cccnc1=O C(=O)(C1=CCN(C(=O)C=C2CCOCC2)C1)NC(c1nn[nH]n1)CC C1(C(N(C(C)C(=O)NOCC2CCCO2)C2CC2)=O)CCCC(C)(C)C1 c1(-c2nc(NC(CC#C)C(C)C)sc2)cc(C)n(CCC)c1C Cc1cc(CC(=O)NC23CC2CN(C(c2coc(CO)c2)=O)C3)cc(F)c1 N1(C(CCOCCOC)=O)CCC(C)(C)C1CC(N1CC(c2nn[nH]n2)C1)=O N1(C2C(NC(CC(=O)NC3CC3)=O)CCC2)CCN(C(=O)CCN2CCCC2)CC1 C(=O)(C#CC1CCC1)NC1C(CCC)CN(C(=O)C(CC2CC2)OC)C1 N1(C(CCCC=C)=O)CCC2CC2(NC(C2CCN(OC)CC2)=O)CC1 C1(C(N(C)Cc2c(C)ccnc2)=O)CCN(C(=O)C(C)CN(C)C)C(C)C1 N1(C(C2CC(=C)C2)=O)CCC(N=[N+]=[N-])(C(N2CCC(c3ncc[nH]3)C2)=O)C1 c1(C(N(C(CCSC)C)C)=O)ccc(CNC(c2ccccc2O)=O)nc1 C(N=c1[nH]c2c(c(=NCC3CCC(C4CC4)O3)[nH]1)CSC2)C1(C(F)F)CC1 C(=O)(CCCCCF)N(C1CCCC1)CCNC(C1CS(=O)(=O)C1)=O S(=O)(=O)(CCCC(=O)NCCN)NCCc1nnn(C(C)(C)C)n1 CC1CCC(CC(=O)NCC(C)N(C(=O)CC(C)n2cccc2)C)C1 C1(NCCC)CCCCC1NC(c1cc[nH]c1)C N1(C(C(C)n2ccnn2)=O)CCC2C(C(N3CC(N(C)C)C(C)(C)C3)=O)C2C1 C1(C(=O)NC(C)CNC(c2ccc(Cn3ccnn3)cc2)=O)CC2CC1CC2O C(=O)(C(CN(C)C)NC(=O)C(=C1CCCCC1)F)NC(C=C)C1CC1 N1(C(C2CN(C(CCOCCOC)=O)CC2(F)F)=O)CC(C)N(C)C(C)C1 N1(C(=O)CN2CCCCC2)CCC(NC(C2(CC3CC3)CC2)=O)C12CC2 C=CCC(C)(CNC(C1CCC(n2cc(C3CC(F)(F)C3)nn2)CC1)=O)CO c1(C(=O)NC2(C)CCC(NC(C3CCS(=O)CC3)=O)CC2)ccc(F)c(C#N)c1 Cn1c(O)nc2cc(C(=O)NC3CCC(NC(C4CC4C#N)=O)C3)ccc12 c1(C(CC(=O)NCCN(C(=O)COCP(C)(C)=O)C(C)C)C)ccc(F)cc1 c1(C(N2CCC(C(C)NC(C3(C(=O)OC)COC3)=O)C2)=O)cnc(O)c(C)c1 C(=O)(C(CC(F)F)N(C(=O)CCN(C)CCO)C)N1CCC(CC(C)C)C1 c1(C(N(CCN(C(CCOCC)=O)C(C)C)C)=O)c(N)cc(F)cc1F N1(C(C(CC)n2ccnc2)=O)CCC(CN(C(=O)CC(C)C2CCCC2)C)CC1 CC1CC(C)N(C(c2ccc(C3CCCCC3)o2)=O)CCN1C(=O)CNC(N)=O C1(NC(C2CCN(C)C2)=O)CN(C(c2cc(C(C)(C)C)n[nH]2)=O)CC2(CCC2)C1 N1(C(C2(CNC(c3cc(Cl)cs3)=O)CCCO2)=O)CCC2(CCCO2)C1 N1(C(C(C)CNC(C2CCCC23CCC3)=O)=O)CCC2(CC1)CC2C#N C=CCCC(C)(C)C(=O)NCC1CC(CNC(C23CCC(C)(CC2)OC3)=O)CO1 N1(C(C#CC2(CC)COC2)=O)CCC2(CC1)CCN(C(c1nc(C)sc1C)=O)C2 N1(C(C)C)CCN(C(=O)CNC(=O)CNC(C2COCCO2)=O)CC1 c1(C(N(c2cccc(CC)c2)C)=O)cc(C#N)n(C)n1 c1(C(N2CCC(N3CC(=O)NCC3)C2)=O)cn2cccc(Cl)c2n1 c1(CC)ccc2occ(C(=O)N(C3CCN(c4nc(C)cc(C)n4)CC3)C)c2c1 CCCC(C(=O)NCCCN(C1CC1)Cc1nnc2ccccn12)C(C)C C1(C)(C(N(CCC2N(C(CCC#CC)=O)CCCC2)C)=O)CC2CCC1C2 N1(C(c2c(OC)ccs2)=O)C2CCC1CC(CNC(c1cc(Br)n[nH]1)=O)C2 C1(NC(=O)OCc2cccc(Cl)c2)CC2(CCN(C(=O)NC3CC3)C2)CO1 C(=O)(CCC(C)S(C)(=O)=O)NC(CCCC)CNC(=O)CCSCC C=Cc1cncc(C(N2CC(C(O)C(=O)NC3CN4CCCC3C4)C2)=O)c1 Cc1cnc(C(=O)NC2CC(C(=O)NC3C=CCCCC3)C2)c(C)c1 C(=O)(CS(=O)C(F)(F)F)N(CCCNC(=O)CCc1cncn1C)C N1(C(C(CCNC(C2CC2C(F)(F)F)=O)OC)=O)CCn2ccnc21 CCCCC(C(=O)N1CC2C(CNC(c3coc(O)n3)=O)C2C1)N(C)C N1(C(C(C2CCCC2)OC)=O)CCC(C2CCCN(CCCCCCO)C2)CC1 C(=O)(C(O)CC(F)F)NCC(COC)NC(c1sccc1OC)=O N1(C(C(C)O)=O)CC2C3CCC(C2C1)N(C(=O)C(c1ccccc1F)C)C3 NS(=O)(=O)C1CCCN(c2ccnc(NC(c3ccccn3)CC3CC3)n2)C1 C(=O)(C1=CCC(C)CC1)N1C(C(=O)OC)(CNC(=O)CC(C)C(=O)OC)C=CC1 C1(O)(CNC(c2nocc2Cl)=O)CCN(C(C2(OCc3ccccc3)CC2)=O)C1 c1(CC2(CNC(=O)Nc3cnn(C(CC)C)c3C)CC2)cc(Cl)ccc1Cl N1(C(C(CC)(C)C(F)F)=O)CC2(C1)CN(C(=O)CC1CCCC1(F)F)CCO2 Cc1cccc(CC(N2CC(CCNC(C3(C)CCOC(C)C3)=O)C2)=O)c1C N1(C(Cc2ncc(C)o2)=O)CCCC2(NC(=O)Cc3ccc(F)cc3)CCCC12 CC1CCN(C(c2cncc(C(C)(F)F)c2)=O)CCN1C(=O)CCOC1CC1 Cc1cccc(CC(=O)NC23CC(C(N4CCC(O)(C(F)(F)F)C4)=O)(C2)C3)n1 C(=O)(C1COc2ccc(F)cc21)NC1CN(C(CC(CC)CC)=O)CC1C C(=O)(C#CC1CCCCC1)NC1C(CC)CN(C(c2coc(C(F)F)n2)=O)CC1 N(C1CCCc2c(F)cc(Cl)cc21)Cc1cccc([N+](=O)[O-])c1Br C=CC(C)(C)CC(=O)NC(C)CCNC(c1ccc(C(F)(F)F)cc1N)=O CCC(C(=O)N(CC(N1CCN(C(C2CCOCC2)=O)CC1)=O)C)C(C)C c1(C(N(CC(CC)NC(=O)C(C)(O)CC(C)C)CC)=O)ccc2oncc2c1 C1(C(C)C(=O)N(C2CCCC2)C)CCN(C(=O)COC2CCCC2)CC1 C(=O)(C(O)CCCNC(=O)C1=NNC(=O)C1)NCC(C)OC C(C(=O)N(O)Cc1cn(C2CCC2F)nn1)NC(COC)=O c1(C(=O)NCCSCCC=C)cccc(CNC(C2CCCN(C)C2)=O)c1 CC(C)CC(C(=O)NCCOC1CN(C(=O)C(C)C(C)O)C1)N1CCCCC1=O N1(C(c2cc(SCC)ncc2)=O)CCN(C(c2nn(C)c(Cl)c2Cl)=O)C(C)C1 c1(C(N(C(c2scc(C(C)=O)c2)=O)CC2NC(=O)NC2=O)=O)ncccc1F c1(NC2CCN(c3c(C(C)C)c(Cl)ncn3)CC2C)ccc([N+](=O)[O-])c(O)n1 C1(C(=O)OC)CS(=O)(=O)C(C)(C)CN1C(C12COCC1CN(C(=O)CC#N)C2)=O C(=O)(C1=C(Cl)CCCC1)N1CC(CC(=O)NC(CCCCC)C)(OC)C1 c1(C(=O)NC2C(CNC(CCNC(=O)NC)=O)C2)ccc(C2CC2)nc1C N1(C(C(CC=C)NC(C)=O)=O)CC2(CC(CNC(=O)C(c3cnn(C)c3)C)C2)C1 C1(CNC(CC(=C)C)=O)CN(C(c2cc(Cl)c(OC)c(Cl)n2)=O)CCC12CCC2 c1(C(=O)NC2CCCN(C(=O)CCNC(c3ccncc3)=O)C2)cccc(=O)o1 Cc1[nH]nc(C(N2CCC(NC(c3ccc(C(F)F)cn3)=O)C2C(C)C)=O)c1Cl N1(C(c2cc(C(C)=O)oc2)=O)CCN(C(c2sccc2C(F)F)=O)CC1C S(=O)(=O)(c1ccc(N(C)CC2CC2)cc1Cl)NC(C)Cn1cccn1 C1(CC(=O)NC2CCCCC2CCO)CCCN(C(=O)C(c2ccccc2)O)C1 N1(C(c2cn(CCC)nc2)=O)CCN(C(=O)Cc2ccc(C)s2)C2CCCCC12 CCCCS(=O)(=O)NCC(=O)NC1CCN(C(=O)C=Cc2cccn2C)C1C CCS(=O)CC(=O)NC(CCNC(C1(COC)CCOCC1)=O)C(C)C c1(CNC(N2C(c3nc(C)[nH]n3)COCC2)=O)ccc2ccncc2c1 C1(NC(c2c(NCC)cccn2)=O)CN(C(C2CCC3CC3CC2)=O)CCC1F c1(C(=O)NCC(CC)NC(c2cc(C(C)C)ccc2F)=O)cnc(O)c(C)c1 c1(C(=O)NCC(CC)NC(c2scnc2C(C)C)=O)cc(F)cc2c1CCC2 CCCC(C)(O)C(=O)NCCOCC(=O)NCC(C)OC c1(C(=O)NC(C2CCCC2)CNC(C2(OC)CCC2)=O)ccc(OC(C)C)cn1 C1(C(N(CCNC(CC2N(C(C)=O)CCC2)=O)C2CC2)=O)CCC(CO)CC1 CCC(C)CC(C)N=c1nc2scnc2c(NCCn2ncc(Br)n2)[nH]1 c1(CC(C(=O)NC2CCC(CC)O2)NC(CCOCCC)=O)cnn(C)c1O N1(C(c2n(COC)ncc2)=O)CCC=C(C(=O)Nc2cnc(Cl)nc2C)C1 C1(CC=C)(NC(=O)CCOC)CCN(C(=O)C=Cc2csc(Br)c2)C1 C(=O)(CCCC(=O)NCC1(C(=O)NCCC2CC(C)C2)CC=CC1)OCC C(CC1c2ccccc2CCN1C(C1CC(C)C1)=O)NC(C(CCC)(C)CC)=O CS(=O)(=O)c1cc(C(=O)Nc2cc(F)c(N3CCCS3(=O)=O)c(F)c2)ccc1Cl c1(CC)nn(C)c(CC(=O)NC(CN(C)C(C2CC(C)(C)C2)=O)CC)c1Cl N1(C(CCCC=C)=O)CCC2CN(C(=O)C#CC3CCOCC3)CCC2C1 CN1CCC(CNC2(C(F)(F)F)CC(F)(F)C2)C1c1ccc(Cl)cc1 c1(COCC)nc(Cl)cc(=NCc2ccc(CNC(=O)C(C)O)cc2)[nH]1 C1(CC)CCCN(C(C2C3CCCOC23)=O)C1C(=O)NC1CCNC(=O)C1 n1(CC(N2CC(NC(c3cc(C(=O)OC)sn3)=O)C(C)C2)=O)nc(C)c(Cl)c1C C1(NC(C(F)=CCC)=O)CC(NC(C2CC3CC(=O)C2C3)=O)C12CCC2 Cc1ccc(C=CC(N2CC3CC(NC(c4snc(Cl)c4Cl)=O)CC3C2)=O)cc1Cl C(C)(CCCN=c1ccc(S(=O)(=O)N2CCCC2)c[nH]1)NC(C(CSC)(C)C)=O C(=O)(C(C)C1=CCCC1)NCCCCCN(C(C(CC=C)C)=O)C c1(NC(c2cnn(C3CCCNC3)c2)=O)ccccc1N1C(=O)C2CSC1C2=O c1(C(=O)NCC2CCCN(C(C(COCC)C)=O)CC2)cccc2[nH]ncc12 c1(-c2cn(C(C)C(=O)NC(Cc3ccccc3)C(=O)O)nn2)ccc(C2CC2)cc1 CC1=C(CNCC2(C(C)C)CC2)S(=O)(=O)CCO1 N1(C(C(C)CC(N)=O)=O)CCCC2(CCCN2C(=O)Cn2cccc(C)c2=O)C1 CC1(N2CCC2)CCC(c2nnnn2C2CCOC2)(NCc2sc(Br)cc2Cl)CC1 c1(OCC)cccc(C(N2CC(NC(c3ccon3)=O)C(n3cccn3)C2)=O)c1 C1(C2CN(C(c3nnccc3C)=O)C2)(NC(C2C(CCC)C2)=O)CC1 C(=O)(CC(C)(O)C=C)N(CCN1CCN(C(C(C=C)OC)=O)CC1)C N1(C(C)=O)CCCC(NC(C2CSCCN2C(=O)CC2CC3(CC3)C2)=O)C1 C1(C(=O)OCC)CC12CCN(C(=O)CN(C)C(=O)NC)CC2 c1(C(=O)NC(CNC(COCCCC#C)=O)(C)CO)ccc2c(c1)CCC(C)N2 c1(C(=O)NC23CC(CNC(C=NOC)=O)(C2)C3)cc(F)c2[nH]nnc2c1 CC(C1=CCN(C)CC1)NC(C1(NC(=O)OC(C)(C)C)CC1C)=O C1(NC(COCC(=O)NC)=O)CCN(C(C2(C#N)CCC2)=O)C1 c1(C(=O)NC2CCC(C(N)=O)C2)ccc(CNC(=O)C(c2ccccc2)O)nc1 Cc1c([N+](=O)[O-])cccc1S(=O)(=O)NC1CS(=O)(=O)C2CNCC12 c1(SC)ncc(Br)c(N2CC3(CN(C(=O)CC4CCC5CC45)C3)C2)n1 C=C(CNC(C1(NC(=O)CNc2ccccn2)CCN(C)C1)=O)C(F)(F)F c1(C(=O)NCCCCNC(=O)Cc2cccc(F)c2F)noc2cc(Cl)ccc12 c1(C(CNC(c2nnn(C)n2)=O)NC(c2cnc(C3CC3)s2)=O)cccc(Cl)c1 c1(Cn2ncc(SCc3n(C(C)C)cnc3)c2)ccc(F)cc1Br c1(OC2(CC(=O)NCC(C)CNC(C3(O)CCSC3)=O)CC2)ccccc1 N#CC1(C(N2CCC(C3CC3)(NC(c3cccc(Cl)c3F)=O)C2)=O)CC2CC2C1 N1(C(CCc2c(C#N)cccc2)=O)CC(NC(c2ccns2)=O)C(C2CC2)C1 c1(C(N(C)CC2CCN(C(CC(C=C)C)=O)C2)=O)ncc(OC)cc1F N1(C(C(C2CCC2)OC)=O)CCCN(C(C2CN3CCCN2CC3)=O)CC1C c1(C(=O)NC(C(C(=O)NCCn2c(C)nc(C)n2)C)C)ccc(C#N)cc1 N1(C(C(C)CC2CC2)=O)CC2CC(C(=O)NC(C34CC(CO3)C4)C)(C2)C1 C1(C2CC2)(NC(c2cnnc(O)c2)=O)CCN(C(c2cc(Cl)c(F)cc2Cl)=O)C1 C#CCCCCCCCCCC(=O)NCC1CCCN1C(c1cnc(Cl)s1)=O C(=O)(C(C(=O)N1CCC(N(C(c2ccc[nH]2)=O)CC)CC1)C(C)(C)C)OCC CC1(CC(=O)NCCOCCNC(C2(F)CCCOC2)=O)CCOCC1 Cc1oc(S(C)(=O)=O)cc1C(N1CC2CC2(NC(=O)CC(C)(O)c2ccccc2)C1)=O O(NC(=O)C(CC(C)C)OC)C(C(=O)OC)CNC(=O)CN(C)C N1(C(C(C(C)C)NC(C2(C#N)CC(C)C2)=O)=O)CC2(C1)CC(C)(O)C2 c1(C(N2CC(CCNC(C3CCC(C)C3)=O)C2)=O)ccc(S(N)(=O)=O)cn1 CCC(CC(=O)N1CCC(C(N2CCC3C(O)CC23)=O)(OC)C1)C(F)F c1(C(C(N2CCCC(CCNC(CS(C)(=O)=O)=O)C2)=O)(F)F)cccc(Cl)c1F N1(C(c2cnc(CCCC)s2)=O)CC2(NC(=O)Cc3ccncc3)CC1C2 CN(C)NC(=O)CCC(=O)NCc1ccsc1C(N1CCC(F)(CO)C1)=O CC1(C)CC(C(N2CC3CC3C3CC23)=O)CN1C(C1CC2C=CC1CC2)=O c1(C(=O)OC)cc(C(=O)N(C)CCN(c2ccccc2)C(C2C3COCC23)=O)cs1 C(=O)(CCCCCNC(C1CCCC1CC)=O)NCC(CC)CCO c1(C(CNC(C2(N)COC2)=O)(F)F)ccccc1 N1(C(C(F)=C(C)C)=O)CC(CNC(=O)C=CI)N2CCC1C2 C1(CN(C)C(C2(C(F)F)CC2)=O)C2CN(C(C3(F)CC=CC3)=O)CC12 Cc1cc(C(=O)NC2CCN(C(c3csc(C(F)F)n3)=O)CC2CO)c(C)cn1 C1(c2cc(NCC)c(O)c(OC)c2)NC(=S)N(C)C(C)=C1C(=O)OC Cc1cc(Br)c(C(=O)NC2CCC(C(=O)NCc3cccc(F)c3)CC2)cc1F C1(CC(=O)N(CCN(C(=O)C=C2CCOCC2)C)C)CCS(=O)(=O)C1 c1(C(=O)NC(C)(C)CNC(=O)C(O)C(C)(C)C)ccc2sccc2c1 C(N=c1cc(C)nc(N(C)Cc2nnc(C)s2)[nH]1)c1c(F)cc(C)cc1F C(=O)(CC(C)(C)CC(F)(F)F)N1CCN(C(C2=NOC(C)C2)=O)C(CF)C1 CCC(C)C(C(=O)N1CC(O)CC1C(N1CC2(C=CCO2)C1)=O)N(C)C C(=O)(CN=c1cc[nH]cc1)NC(CC)CNC(c1ccc(Cl)cc1OC(F)F)=O C1(C(=O)NC2CCN(C(Cc3nnc(C)s3)=O)C2C2CC2)CCn2nccc2C1 CCCCCCCCNS(=O)(=O)CC1CCC(C)CO1 N1(C(c2cc(SC)oc2C)=O)CCOC2CCN(C(c3ccc(CO)s3)=O)CC12 N1(C(CSCC(C)=O)=O)CCOCC(NC(=O)C(c2ccc(F)cc2)(F)F)C1 N1(C(C2=C(C)CCC2)=O)CC2(CC(NC(=O)CCC(C)N(C)C)CO2)C1 C(=O)(C1=C(C)CC(C)(C)CC1)NCC1(NC(c2c(CC(=O)OC)occ2)=O)CC1 c1(C(N2C(C(=O)NC3CCOCC3F)(CC)CCC2)=O)cc(C)c(C)nn1 Cc1cc(-c2cncc(C(N3CC4C(C3)C4(F)F)=O)n2)cc(F)c1 N1(C(C2(NC(CCC(C)=O)=O)CCN(C)C2)=O)CC(C)OCC(C)(C)C1 C(=O)(CCCC(C)NC(=O)C(C1CC1)SC)NC(c1nc(CC)[nH]n1)C C(C)(C)(CC(C)(C)O)NC(C1CN(C(Cc2c(C)nn(C)c2)=O)CC1F)=O N1(C(c2nc(C)c(Br)cc2)=O)CC2(CCC(C(=O)NCC3(C)CC3)O2)C1 C1(C(=O)OCCN2CC(C)CC(C)C2)CC2CCCC(C1)C2=O C1(C(N2CC(C)(CCO)C2)=O)(OC)CCN(C(c2csc(C)n2)=O)C1 C1(COC)CN(C(c2cc(C)n(C(F)F)n2)=O)CCN1C(=O)C1=COCCC1 C(=O)(C1COc2ccc(Cl)cc21)NCC1CCCC2(CN(C(C(C)CF)=O)C2)O1 c1(SCCC(=O)NC2CC(NC(CC3(OC)CCC3)=O)C2)nnnn1C Cc1cccc(C=CC(N2CC3(CC3)CC2C(=O)NCc2ccc(Cl)nc2)=O)c1 c1(CNC(N2CCC(Cc3c(Cl)ccc(OC)c3)CC2)=O)ccc(O)c(C#N)c1 C1(C)(COC)CCC(NCC(=O)N(c2ccc(C)c(F)c2)CC2CCCO2)CC1 C1(NC(C(COC)C)=O)CN(C(C23CC(CO)(C2)C3)=O)CC1SC N1(C(C2CC(C)(CC)C2)=O)CC=CC(NC(c2oncc2C)=O)C1 O=C(C1=CCCN(C(=O)CCc2ccncn2)C1)N1CCOCC1CCO C1(CC)CN(C(=O)C(O)C2CC2)CCC1CNC(c1c(C)cccc1O)=O C(C)(C)(CCCC(=O)NC(C)C(C)CO)NC(CCNC(C)=O)=O c1(C(=O)NCC2CC(NC(=O)CCF)C23CCC3)cc(F)c(O)cc1Br C(=O)(CC(C)C(C)(C)NC(=O)CN1CCSCC1)NC(CC)CCCO Cc1cccc(C)c1N(CC(C1CCN(C(=O)Nc2nccs2)CC1)C)C(C)C C1(NC(C2C(c3n(C)ncc3)C2)=O)CCN(C(c2ncc[nH]c2=O)=O)CC1CO CC1(C)C(CNC(C2(n3cc(COC(=N)O)nn3)CCOCC2)=O)C1C#N c1(COC)ccsc1C(=O)NC(CNC(=O)Cc1csnc1C)CCOC c1(C(=O)NCC(c2cccc(Cl)c2)F)cc(Br)c2ccccc2c1 c1(C(N(C)CC2C3CN(C(CN(CC)CC)=O)CC32)=O)cc(OC)c(F)c(F)c1 Nc1ccc(O)c(C(=O)NCC2CCCN(C(=O)Cn3cc(Cl)cn3)C2)c1 c1(C(N(C)CC2(CNC(=O)COCc3ncnn3C)CC2)=O)cccnc1S c1(C(N2CC(O)(CNC(=O)CCC(F)F)C2)=O)cncc(O)c1Cl c1(C(C(=O)NCCN(C(CC(C)n2cccn2)=O)CC(C)O)=O)ccc(O)cc1 CC(C(C(=O)N(CCCF)C)NC(=O)OC(C)(C)C)c1ccccc1 c1(C(=O)NCCN(C(C2C(C=C)OCC2)=O)C2CC2)nccc(OC)c1OC C1(N(CCNC(c2ccc(C(=O)O)o2)=O)CC)CCCN(C)C1=O C(=O)(C(O)CCCNC(=O)Cc1cccs1)N(C)Cc1c(C)occ1 C1(=CC(=O)NC2CC(C)N(C(=O)CCCc3cncs3)C2)CCC(C)(C)CC1 C(=O)(CS(=O)(=O)Cc1cccs1)NCC1(CNC(C(CSC)(F)F)=O)CC1 C1(C(N(CCNC(c2n(CC)c(O)nc2)=O)C)=O)CCC(N=[N+]=[N-])CC1 C1(CNC(=O)Cc2nc(CCCO)n[nH]2)CCCCN(C(c2cc(Cl)ccn2)=O)C1 N1(C(c2c(Cl)cc(C)s2)=O)CC2(CCOCC2)CC1CNC(c1csc(O)n1)=O C(=O)(C1=NOC(C)C1C)NCC1COCCN(C(C2(C(=O)NC)CC2)=O)C1 C(=O)(C(C)(C)CN(C)C)NCCC(C)(C)NC(CCNC(C)=O)=O.C1CSC1 Cc1cc(C(=O)N(C2CCN(C(=O)C(C)C(C)C)C2)CCO)cc(C)n1 C1(C(N(CCN(C(=O)C(C)Cn2ccnc2)CC)CC)=O)OCC2CCCCC12 c1(NC)cccc(C(=O)NCC2CC(NC(=O)C(C)NC(c3ccco3)=O)C2)c1 N1(C(c2cnc(C)o2)=O)CCC2(CC1)CC2NC(=O)CC1CC2(CC2)CO1 Cc1cc(C(=O)NC(C(C)NC(c2ccsc2C(F)(F)F)=O)C(C)C)c(O)nn1 N1(C(c2cc(C)nc(O)c2)=O)CCC12CCCN(C(c1cnc(Cl)s1)=O)C2 C1(CCNC(CC(=C=C)C)=O)CCN(C(c2nccc3[nH]ccc23)=O)CC1(F)F N1(S(CC)(=O)=O)CCC(C(=O)N(C2CCCN(CCS(=O)(=O)CC)C2)C)CC1 c1(C(N2CCN(C(C3(C)CC3Br)=O)CC2)=O)cccc(C(F)F)c1F c1(CC)cccc2c(C(=O)NCC3(NC(=O)C4=CCCOC4)CCCC3)c[nH]c12 c1(OC)cccc(CCC(=O)NC2CCCCC2N(C(=O)C#CC2CC2)C)c1 c1(C(=O)NC(COC)CC(=O)NCCCN2CCCCC2)cc2cccnn2c1 C1(CNC(c2cnn(C)n2)=O)COCCN(C(=O)CC2(C#N)CCC2)C1 C1(C(N(C(C(C)SC)C)C)=O)COCCC1NC(=O)C(C(C)C)NC=O Cc1nc(O)[nH]c1C(=O)NCC(C1CCC1)NC(=O)C(F)Cc1ccccc1 Nc1sc2cccnc2c1NCCCCc1ccccc1F c1(C(N2CCC(NC(CCC(C)SC)=O)C2C)=O)cn2nc(C)cc2[nH]c1=O N1(C(CC2N(C)CCOC2)=O)CC2CCC(C1)N2C(=O)Cc1c[nH]nc1O N1(C(c2c(C)ncnc2)=O)CC(NC(=O)C=Cc2cn[nH]c2)CC12CCCOC2 c1(NC(C(=O)N(C2C(C)CCC2)C)=O)ccc2oc(CC(F)(F)F)nc2c1 C(C(C)(C)C(=O)N1CC(O)(C(F)C(N2CC(C)(C)C2C2CC2)=O)C1)SC Cn1c(SCCO)nnc1C1CCCO1.C1CCN1C(=O)C=CC(N)=O Cc1cccc2c(C(N3CC4CC(NC(=O)C5=CCCOC5)C(C4)C3)=O)n[nH]c12 N1(C(COCCCOC)=O)CCCCC1C(=O)NCCc1ccnc(C)c1 N1(C(C2(CC=C)CCOCC2)=O)CCC2CN(C(=O)CCCC#N)CC2C1 CCCCC(O)CCC(=O)NCC=C1CCN(C(C2(C)CC(F)C2)=O)CC1 N1(C(COCC=C)=O)C2CCC1CC(O)(CNC(C1C3CNC(=O)C13)=O)C2 C(N=c1[nH]c(N2Cc3c[nH]nc3C2)nc2c1CCC2)c1c(CC)n[nH]c1 c1(C(=O)NCCCCC#C)cc2ncc(-c3cnc(C)c(C)c3)cc2[nH]1 C1(NC(c2nc(CC)sc2)=O)CN(C(=O)C(C)CC2CCC2)C(C)(C)C1 O=C1OCCN(Cc2ccc(-c3ccc(C(=O)O)o3)cc2)C1CCO N1(C(c2ccc(C(=O)OC)s2)=O)CCCC(F)(CNC(C2COC(C)C2)=O)C1 CC1(NC(c2nocc2Br)=O)CCN(C(C2COCCO2)=O)CC1 N1(C(c2c(CC(C)C)onc2)=O)CCC(NC(c2cc(CC(C)C)on2)=O)CC1 c1(C(=O)NC2CC(CNC(c3cncs3)=O)C23CCC3)n[nH]c2ccc(Cl)cc12 C1(C(=O)NC(CN(C(CCC2C(C)=NOC2=O)=O)C)C)CCc2nn[nH]c2C1 C1(NC(C=CC(C)C)=O)CS(=O)(=O)CC1NC(=O)CSC1CC1 Cc1nc(C(=O)NC2(C)CCN(C(c3ccc4c(c3)CC4)=O)C2)ccc1[N+](=O)[O-] C1(CC(=O)NCC(C)CC2CCCC2)CCCCC1 C1(NC(CCCCC=C)=O)CC2(C1)CC1(CC(NC(C3(C#N)CCOC3)=O)C1)C2 C1(OC)CN(C(=O)C(C)O)CCC1NC(c1sc(Cl)c(Cl)c1C)=O C(=O)(CC(C)CNC(=O)C(=O)NC(C(C)C)C1CCC1)NC c1(C(=O)NCC(CC)(C)NC(=O)C(N2CCN(C)CC2)C)cnc2cc[nH]c2c1 C1(NC(C23CC(C)C2C3)=O)CCN(CC(F)(F)F)C1=O N1(C(c2cc(CC)nn2C)=O)CCC(F)CC1C(=O)NCC1(C)CC2(CC2)C1 C(=O)(C(CC)C(C)(C)CC)NCCN(CCC)C(c1cc(C)n(C2CC2)n1)=O C(C(=O)N1CC2CC(N(C(=O)CCc3cccs3)C)C1C2)(C(C)(C)C)SC N1(C(C(C2CCC2)OCC)=O)CC(O)(CCC2(CC)CCC2)C1.C1(=O)C(CC)N1 c1(OC)ccc(CN=C(NCC(F)F)NCC2(c3ccncc3Cl)CC2)cc1 c1(C(=O)NCC#CC(=O)NCC#CCOC)cc2cnccc2[nH]1 C(=O)(CC(O)CNC(=O)Cc1cnoc1)NCC(C1CCC1)OC C(CC(F)F)(C(=O)NCc1ccnn1CC)NC(c1c(C)nc(CC)o1)=O C1(NC(c2ccc(CN(CC)CC)cc2)=O)CC(C)CN(C(=O)C=C2CC2)C1 N1(C(COCCNC(CC)=O)=O)CCN(CC2CCCO2)CC1 n1(CC(N2C(CNC(c3c(C)cc(C)s3)=O)C(C)CC2)=O)cnc([N+](=O)[O-])n1 C(CNC(=O)C(COC1COC1)OC)(CC)(CC)NC(CC1(CC)CCCC1)=O c1(C(C)NCC(c2ccccc2F)F)cccc(F)c1 C1(C(=O)NCc2cccc(C(=O)NC3(CC)CCC3)n2)CC2(CCO1)CC2 Cc1c(C(=O)NC2CC(N(C)C(C3SC4C=CC3CC4)=O)C2)[nH]c2ccccc12 N1(C(CCC2N(C(CNC(C(C)(C)C)=O)=O)CCC2)=O)CCCC(O)CC1 c1(C(N(CC(C)(C)CNC(=O)C(N)=O)C)=O)ccc(=O)n(-c2cnn(C)c2)c1 N1(CC(=O)N(C(C)CNC(c2cnc[nH]2)=O)CC)CCCS1(=O)=O C1(CC=C)(C(=O)N(C)CCOCCN(C)C)CCCN1C(=O)CCO.C1CC1 O(C1c2ccccc2C2CC1C2)C(c1ccn2ncccc12)=O N1(C(c2occ(C(=O)OC)c2)=O)CC(NC(=O)C(C2(O)CCCC2)F)C2(CC2)C1 C12(C(N3CC(NC(COCC#C)=O)C(C)CC3)=O)CCC(C(=O)OC)(CC1)CC2 C1(CC(N2C(C)CCC(CNC(c3csc(O)n3)=O)C2)=O)Cc2ccccc2N1 N1(C(C(C)n2cnnn2)=O)CC2CCCN(C(=O)CCC3CCC(=O)C3)C2C1 CCC(C)C(O)C(=O)NCC1CC(NC(C2(c3ccc(C)nc3)CC2)=O)C(O)C1 C12(NC(=O)CCOC3CC3)CCC(CC1NC(C1CCS(=O)(=O)N1)=O)C2 N1(C(C(CC)n2cncn2)=O)CCN(C(=O)Cc2cnsc2)C(C(C)C)C1 N#CC1(c2cn(CCCC(=O)NCCCC(=O)N3CCCC3)nn2)CCCC1 c1(C(=O)NCCN(C(C(C)N(CC)CC)=O)C(C)C)cscc1S(C)(=O)=O c1(C(C(=O)NC(CC)C)N(CCCCOC)C)cnn(C2CCCC2)c1 CCCCC(C(=O)N(CCCCCNC(C1OCCN(C)C1=O)=O)C)C(C)C N1(C(C2C(C=C)OCC2)=O)CC(NC(c2cccc(F)c2)=O)CC1(C)C C(CNC(c1oc(Br)nc1C(F)F)=O)(C(C)C(C)C)NC(CC=CC)=O c1(C(N(C)CC2CN(C(C3C(C)CCC3)=O)C2)=O)cc(F)cnc1O N1(C(C(C)S(C)(=O)=O)=O)CCCC(C2CCCN(C(C3COC(=O)O3)=O)C2)C1 C(N=c1[nH]c(N2CCC3CC3C2)nc2cccnc12)c1c(F)ccc(N)c1 C1(CNC(C2CCOC2)=O)CCCCN1C(c1c[nH]nc1-c1cccs1)=O N1(C(c2c(NC)cccc2)=O)C(C(=O)Nc2ccc(O)c(F)c2)CC2CCCC12 C1(C(=O)NC(c2nnnn2C)C)CN(C(C2CCC(C)(C)C2)=O)CC1(F)F CC(=O)CCCC(=O)N1CC(CNC(c2cnccc2N(C)C)=O)CC1C C(=O)(C1CCc2nccn21)N1CCCC(CNC(c2c(N)nccn2)=O)(CO)C1 Cc1noc2ncnc(N3CC(NC(c4n[nH]cc4C4CCC4)=O)CCC3C)c12 C(=O)(C1=C(F)CN(C(c2ncc[nH]2)=O)CC1)NC(C)(C)CC(N)=O N1(C(C(c2c(C)n[nH]c2C)C)=O)CCN(C(=O)CC(C2CC2)C2CC2)CC(O)C1 c1(CC)onc(C)c1C(=O)NC(CCc1ccccc1)C(C)NC(=O)CCC#N c1(C(=O)NCC2CC(OC)CN2C(C2(F)CCCN(C)C2)=O)cncc(F)c1Cl c1(NC(c2nc(-c3cccnc3-c3nn[nH]n3)cs2)=O)cc(F)c(F)c(F)c1 C(CCCC(=O)NCc1ccc(C(=O)NC2(CO)CCC(C)C2)cc1)SC c1(OC)cc(CC(=O)NCCC2CC(NC(c3c(C)csc3Cl)=O)C2)ccc1C Cc1csc(=O)n1CC(N1CCCC(C2CCCCN2C(c2cnn[nH]2)=O)C1)=O O=C1NC2CN(C(=O)COC3CCN(C(=O)CCc4cccnc4)C3)CC2O1 Cc1ccc(C(N2CCC(C(F)(F)F)CC2C)=O)c(C2CC2)n1 O=C(C#CC1CCOC1)NC1CC(CNC(C2CC2C(F)F)=O)C1 CN1CC2CCCC(C1)N2C(=O)CSCCNC(c1c[nH]c(=N)o1)=O c1(C(=O)NCC2N(C(c3c(CC)[nH]cc3)=O)CCC2C)ccc(N=[N+]=[N-])cc1 c1(C(N2CCN(C(c3c(C)coc3)=O)C(C(C)C)C2)=O)csc(=NC2CC2)[nH]1 Nc1cc(N2CCS(=O)CC2)ccc1-n1cc(-c2ccc(C(F)(F)F)cc2)nn1 C(=O)(C(O)CCCc1ccccc1)NC1(CNC(C2C(C(=O)OC)C2)=O)CC1 C12(C(=O)NCC3(NC(CS(CC)=O)=O)CCCCC3)CC(CO)(C1)OC2C CC1(O)CON(C(=O)C2CCC3(CC3)NC2)C1 C1(c2n(CCSC)nnn2)(NCC2CC23CCCCC3)CCC(F)(F)CC1 c1(C(N(CCCNC(CC2CC(C(C)C)OCC2)=O)C)=O)cnn2ccccc12 c1(N2CCC(OCC=C)CC2)nc(N(C)C)nc(N2CC=CC(OC)C2)n1 c1(C(N2CC=C(CNC(C3C(CC)OCC3)=O)CC2)=O)cc(C)c(Cl)cc1C CCC(C(=O)NCC1(C)CCCN1C(c1cc(O)ccc1C)=O)C(C)C CCC(CNC(=O)C(=O)NCCCc1ccccc1)C(=O)O c1(C(N(CCCCCCNC(C2CC(OC)C2)=O)C)=O)ccc(C2CC2)c(C)c1 C1(F)(C(=O)NC2CCCN(C(c3n(C)nc(O)c3)=O)C2)CC12CCCCC2 N1(C(c2n(CCOC)ncc2)=O)CC(CNC(c2ccn(C)c2)=O)C2(CC2)C1 Cc1ccc(C(CN(C)C)NC(=O)NCCc2nnc3n2CCC3)cc1F Cc1cc(N2CCSCC2)ccc1NC(C1(C)COCCO1)=O N1(C(CC=CC)=O)CCCC(C2CCN(C(=O)C(C(C)C)SCC)CC2)C1 c1(CNC(=O)CC2CCCN2C(=O)CC2CNC2)ccc(C(F)(F)F)cn1 c1(C(=O)NCCCCCNC(C(C(C)O)C)=O)nn(C)c2ccccc12 CCC(CC)CC(=O)NC1CCC(CNC(C23CC(C)(CCO2)C3)=O)C1 C1(C(=O)NCC2(C)C(C)CN(C(CC(CC)CC)=O)C2)CCC(C2CC2)CC1 CC(CNC(c1cccc(C2CC2)c1)=O)CN=c1cc(C(F)F)c([N+](=O)[O-])c[nH]1 Cc1c(NC(=O)C(C2CCC2)NC(c2cnn(CC3CC3)c2)=O)cnn1CCO CCC(CC)CC(F)C(=O)NC(Cc1ccco1)C(=O)NC1C(C)C1C CCCC(CC)C(=O)NC1CCCC1NC(c1ccc(C(C)=O)cc1)=O CN1CCN(C(C2CC3(CCC3O)C2)=O)C(CNC(=O)CN(C)S(N)(=O)=O)C1 C(=O)(CCC1=CCCCC1)N1CC(C)(CO)C(O)CC1.C12CCN(CC1)C2=O C1(n2cc(C3(C)CCN(C(C4CCOC4(C)C)=O)C3)nn2)(CC)CCOCC1 Cc1c(Cl)sc(Cl)c1C(=O)NC(C)CCNC(=O)C(O)C(C)(C)C CC1(P(C)(C)=O)CCCN1C(=O)C(c1cccnc1)Oc1ccccc1F c1(C(N2C(C(=O)Nc3c(C(N)=O)cccn3)CC2)=O)ccc(Cl)cc1Br C(c1ccc(C#N)cc1)=CC(N1CC(CNC(CC(CCC)C)=O)C2(C1)CC2)=O c1(C(=O)NC2C(NC(C3N(C(CCC)=O)CSC3)=O)CCC2)cccc(CF)c1 C#CC1(O)CCCN(C(=O)CC=CCNC(C23CCCCC2C3)=O)C1 c1(C2CCN(C(C(CF)(CF)NC(=O)OC)=O)CC2)cccc(OC)c1 N1(C(CC(C(C)C)C)=O)CC(C)CN(C(c2cc3c(nc2O)CCC3)=O)CC1C c1(C(N(C2CCN(C(=O)CC34CCCC3C4)CC2)CCC)=O)cncc(SC)c1 C1(SC)CCCC(NC(=O)C(CO)NC(c2cnnc(C)c2)=O)C1 C1(NC(C(F)=CC)=O)COCC1NC(c1scnc1C1CCCC1)=O N1(C(c2cnn(CC)c2C)C(=O)NC2CCOC2)CCNC(=O)C(F)(F)C1 Cc1cc(Cl)ccc1NC(=O)OC(C)C(=O)N(C(C)CN(C(=O)CN(C)C)C)C c1(C(=O)OCC)cnc2c(C)cc(C)cc2c1N1CCN(CC(=O)NCC)CC1 C=CC(CC)CC(=O)N1CCN(C(c2cc(Br)cnc2C)=O)C(CC)C1 C(C(CO)C(F)(F)F)NC(COC(C)(C)CNC(=O)CC1CCCC(=O)N1)=O C1(CNC(c2c(C)ncs2)=O)C2CC1N(C(c1nn(C)cc1Cl)=O)C2 C1(COC)CCN(CCNC(c2csc(CN)c2)=O)CC1 C1(C(=O)NCC2CC(CN=[N+]=[N-])C2)(CNC(c2cccnc2O)=O)CC12CCC2 Cc1cn2c(=O)c(-c3nc(-c4cncnc4)nn3-c3cccnc3)cnc2s1 C1(C(=O)NC(CC)CN(C)C(c2cc(C)c[nH]2)=O)CC2(C1)C(C(=O)OC)C2(F)F N1(C(C=C(C)C)=O)CC(NC(c2nn(C)c3c2COCC3)=O)CC12CCOCC2 N1(C(Cc2cc(C)sc2)=O)CC2CC(C(=O)NCCn3ccccc3=O)(C2)C1 N1(C(C2(NC(C)=O)CCC2)=O)CC(NC(c2c(C(F)(F)F)coc2C)=O)C(C)C1 C=CC1(CC(=O)NCCn2ccnc2CNC(N)=O)CN(C(=O)CCSC)C1 C(C(C(C)(C)C)NC(c1ccnn1C1CCCC1)=O)NC(C(Br)=C(C)C)=O c1(C(N2CCN(C(c3c(C)nco3)=O)CC2C(C)C)=O)ccc2c(c1)nnn2C CC1CCN(C(=O)C(CC(N)=O)NC(C2CC=CCO2)=O)CCS1 Cc1ccc(OCCC(=O)N(CC(O)CN2CCOCC2)C)cc1C C(=O)(CC(F)(F)CC)N(C1(C(=O)NC(CC#C)CO)CC1)C c1(CC(=O)NCC(CCNC(c2ccc(C#N)s2)=O)O)ccc2cnccc2c1 C1(NC(CN(CC(C)C)CC)=O)CC2(C1)CN(C(=O)C(C(C)C)OC)C2 Cc1cc(C(N2CC(c3cn(-c4cncc(Cl)c4)nn3)C2)=O)nn1CC1CC1 N1(C(C2(C)N(C(CC(C)(C)OC)=O)CCC2)=O)CCCC(C)C1CO C(C(=O)N(CCCCCCNC(=O)Cc1cnn(C)c1)C)(C(C)C)OCC N1(C(c2nn(C)c(O)c2)=O)CCC(C(F)(F)F)C(NC(=O)C(C2CC2)C2CC2)C1 CC(C(=O)NCC(O)C(=O)NCC1CCCC1(C)C)C(F)F c1(C(=O)NC2C(NC(c3cn(CC)nc3C(C)C)=O)C2)cccc2c1OCC2 n1(CC(=O)NCCN(C(=O)C(C)(F)C(=O)OC)CC)cnc([N+](=O)[O-])n1 C1(CNC(C(F)=CCC)=O)CCCCN1C(c1ccc(C2(OC)CCC2)cc1)=O c1(CC)nc(O)c(C(N2CCN(C(=O)CC3CC(F)C3)CC(O)C2)=O)cc1C CCC(CS(C)(=O)=O)N=c1nc2c(cnn2C)c(NCCOCC2CCOC2)[nH]1 C1(CNC(C(=O)NCC)=O)CCC12CN(C(c1ccc(OC)cn1)=O)C2 c1(NC(c2c(C)cc(CNC(=O)CCc3ccccn3)o2)=O)cccc(Cl)c1C C(=O)(CC(CC)CCCC)NCC(CC=C)NC(c1snnc1C1CC1)=O c1(C(=O)NC(C2CCN(C(CC3(C(=O)OC)CC3)=O)C2)C)c(OC)ccnc1F Cc1ccnc(C(=O)NCCCNC(c2cccc(-c3cccc(C)c3)c2)=O)n1 N1(C(COCCNC(C#CC2(C)COC2)=O)=O)CCN2CCOCC2C1 C1(Cn2cc(C(C(=O)OCC)(F)F)nn2)CN(C(=O)C(C)(C)C#N)CCO1 Cc1cc(C(F)(F)F)n2c(NC(=O)CN3CC4C5C=CC(C5)C4C3)nnc2n1 C=CC1(C(=O)N(C)CC2COC(=O)N2)CCN(C(c2cc(C)co2)=O)C1 CON1CCC(C(=O)NC(C)(C)COCCCNC(=O)CCC2CCCC2)CC1 c1(C(CC(=O)N(CC(C)NC(=O)C(O)CF)C)NC(C)=O)ccc(Br)cc1 N1(C(Cc2cccc(C)c2)=O)CC(O)C(O)C1CNC(C1(C)CCN(C)CC1)=O C1(OC(=O)NC2C=CC(CN(CCC)CCO)C2)(OC(C)(C)C)CCCC(C)C1 C1(NC(C=C(C)C(=O)O)=O)C2COCC1CN(C(C1CC(N)C1)=O)C2 CC(C(=O)NC1CC2CC1N(C(=O)Cn1cccnc1=O)C2)P(C)(C)=O C1(CC)(NC(C2CC(NC(=O)CP(C)(C)=O)C2(C)C)=O)CCCCCC1 C(=O)(C#CC1CCOC1)NCCCN(C(CC1N(C(C)=O)CCC1)=O)C c1(C(=O)OC)c[nH][nH]c1=NC(=O)C1(O)CCN(C(c2ccc(C)cc2OC)=O)C1 C1(CNC(C2C(C)C2)=O)CN(C(=O)Cc2cccc(F)c2)CCC1C(F)(F)F C1(OC)CC(CNC(=O)CN(C)C)N(C(C2CCCC2C)=O)C1 c1(C(CNC(C2SC3C=CC2CC3)=O)NC(C(CC=C)C)=O)cc(F)cc(Cl)c1 C(=O)(CN=c1cc[nH]cc1)NC(C(=O)N(CCCF)CC)c1ccco1 N1(C(C)=O)CC2CCCC(NC(=O)C(C)NC(=O)O)C2C1.C(CNC(C)=O)OC N1(CCNC(C2(OC)CCC2)=O)CCC(NC(c2cc(C#N)on2)=O)CC1 Cc1ccc(CC(=O)NC2CCCN(C(c3c[nH]c(Br)c3)=O)C2C)cc1O N1(C(c2cc(C)ns2)=O)CC(C(=O)NC2CC2c2ccnn2C)CC12CCC2 C(=O)(C(CCS(N)(=O)=O)NCc1ccccc1N)OC c1(C(=O)NCC(C)CNC(=O)C(c2ccc(F)cc2)CO)cccc2cnsc12 C=CCC(C)(C)CC(=O)NCC1CN(C(c2cccc3nsnc23)=O)C2CC12 C12(C(=O)OC)CCNC1CN(C(c1ccc(OCCCOCC(C)C)cc1)=O)C2 CCCC(C)C(=O)NCc1ccc(C(=O)NC2CC(C)(C(N)=O)C2)nc1 C(=O)(C(O)CC(F)(F)F)N1CCCC(CCCCNC(C(=O)NC(C)C)=O)C1 N1(C(C(C)OC)=O)CCCC(C)(CNC(=O)CCn2nc(C)nc2C)C1 c1(N(CCC)C(C)=O)cc(C(=O)Oc2ccc(Cl)cc2)ccc1C#N c1(CN2CCCC(CC(N3CCCN(C4CC4)CC3)=O)C2)ccc(F)cc1F c1(C(=O)NCC2(O)CN(C(CC(C(C)C)(F)F)=O)C2)nnc2ccccc2c1N S(=O)(=O)(c1ccc(NCCCn2nc(C)cc2C)c(Cl)c1)NCC(CC)(C)OC C1(NC(c2c(CC)ccs2)=O)CN(C(c2cocc2Br)=O)CC2(CC2)C1 c1(NC(C2CN(Cc3c(C)ccc(O)c3)C2)=O)ccc(C(F)(F)F)c(C#N)c1 C1(C(=O)NCC2CN(C(C(CC)=CC)=O)CC2C)(OCC)CCCCCC1 c1(C(=O)NCC#CCNC(C2(O)CCC(CC)C2)=O)ncc(N)nc1C Cc1cnc(C)c(C(=O)NCCC2(C)CCN(C(c3cc4n(n3)CCC4)=O)C2)c1 c1(N2CCC(NC(CC)=O)C(O)C2)nc2cc(F)ccc2o1 C(=O)(C1=NNC(=O)CC1)NCC1CC(NC(=O)C#CC2CC2)C12CCC2 N1(C(C(CC#C)C)=O)CCCCC(CNC(=O)CCC(=O)c2ccncc2)C1 N1(C(C(C)SCC)=O)CCC(C(=O)NC2(c3ncc[nH]3)CC2)(OC)C1 C(=O)(C#CC1CCCO1)NC1(CC=C)CCN(C(=O)CC(C(=C)C)OCC)CC1 C(C(CC(C)C)C(=O)NC1CC(CCNC(=O)CCCC(F)(F)F)C1)OC C(CCCC(=O)NCC(C)(C)OCC(N1CCC(O)(CC(C)C)C1)=O)SC CC1(C)CCC12CCN(C(=O)Nc1ncc(C(N)=O)s1)C2 c1(C(=O)NCC(O)C(=O)NCCCc2ncco2)coc2ccccc12 N1(C(C(C(C)C)C)=O)CC2(C=C(C(=O)NCC3(CCCO)CC3)CO2)C1 c1(CC(=O)NCC(CN(C(=O)COc2ccc(F)cc2)C)O)nc([N+](=O)[O-])n[nH]1 Cc1nc(NC(C)C(C2CCCCC2)NC(c2cocc2C)=O)c2ccsc2n1 C(=O)(CC1OCCc2ccccc21)NC1(CN(C(c2nc(C)oc2C)=O)C)CC1 C(CC(C(C)(C)C)NC(=O)CC(CC)CC)N(C(C(CC=C)OC)=O)C C(=O)(C(F)(F)C(F)(F)F)NC1CCC(NC(=O)Cn2cncn2)CC1 C(=O)(CCCCCC(CC)OC(C)(C)C)NC1CN(C(=O)OCC)C(C)(C)C1 C1(CC(=O)NCCC=CCCC)CCCN(C(=O)CN2CC(=O)NC2=O)CC1 N1(C(c2c(C)n(C)nn2)=O)CCC2(CC1)CCN(C(C1CCC(F)CC1)=O)CC2 c1(C2CCN(C(=O)NC3C(c4cccc(C)c4)C3)C2C)ccc(C#N)cc1 c1(C(=O)NC(C)CNC(=O)C(=O)N(C)C)ccc2c(c1)N(C)CCO2 c1(NC(C2C3CN(C(C(CC)O)=O)CC32)=O)ccc(C)c(OC(F)(F)F)c1 C(=O)(CCC(=O)NC1CCCC(NC(=O)CC2(O)CC2)C1)N(C)C C1(SCC(=O)Nc2c(C(=O)OCC)c(C3CC3)cs2)CCCC(C)(C)C1 C1(CNC(COCCC#C)=O)COCCN1C(=O)C(c1ccc(Cl)cc1)CC S(=O)(=O)(c1ccc(C#N)c(NC(C)CS(C)(=O)=O)c1)NCCCOC(C)C c1(C(=O)NC(C)C(F)(F)C(F)(F)F)ccc2c(c1)CCC2N C=CCC(C)(C)C(=O)NC1CN(c2ncc(C(=O)OC)cc2C)CCC1C c1(C(=O)NC(CN(CCOCC)C)C)ccc(Oc2ccccc2)cc1 c1(OC)cc(C(=O)NC2(C)CCN(C(=O)C=CS(C)=O)C2)cc([N+](=O)[O-])c1 C(=O)(C(COC)CC(C)C)NCCN(CCC)C(c1ccc(-c2ccco2)s1)=O c1(C(=O)NC(C(C)NC(Cn2ncc(C)c2)=O)CO)ccc2ccccc2c1O N1(C(CC(C(F)F)NC(c2ccc(C)[nH]2)=O)=O)CCc2ccc(O)cc21 N1(C(C2CCCN(Cc3cc(Br)ccc3Cl)CC2)=O)CCc2nc[nH]c2C1 C1(C(=O)NC2CC(C)N(C(C3CC(C)(O)C3)=O)CC2)CCc2ccccc2CC1 c1(C(N2CCCC2CNC(=O)NC(C)(C)C)C(=O)NCC)cccnc1C N1(C(c2ccc(C)nc2C)=O)CCC(C2(NC(C3CN4CCN3CC4)=O)CC2)C1 N1(C(COCCC#C)=O)CCC(O)(CNC(C2(C(C)(F)F)CCOCC2)=O)C1 C(=O)(C(F)(F)C(C)(C)O)NCCCCN(C)C(c1cccc(F)c1Cl)=O c1(CS(=O)(=O)NCc2ccc(-c3nc(C4CC4)ns3)nc2)csc2ccccc12 C12(C(N(CCN(C(=O)COCC3CCOC3)C)C)=O)CCN(CC1)CC2 c1(C(=O)NCCCCC(C)NC(=O)CN2CCCCC2)coc2c1C(=O)CCC2 C(N=c1ccnc(C)[nH]1)C12OCC(CNC(C3(CC)CC3)=O)(C1)C2 CC1(NC(=O)CC(O)CNC(C2CCCCO2)=O)CC2(CCC2)C1 CC(C)(CCC#N)C(=O)NC1CCC(CC(N2CCSC3CCC23)=O)C1 C1(NC2C(OC)COC2)C(NC(=O)OC(C)(C)C)CCCC1C N1(C(C(C)OC)=O)CCC(NC(C2CCCCN2C)=O)C1C1CC1 c1(NC2CCN(C(=O)NCCC(COC)(C)O)CC2)cc(C)cc(C)c1 c1(-c2ccc(C(=O)NC(C(C)(C3CC3)OC)C)s2)ccc(F)cc1F C1(CNC(C2C(C)OCCO2)=O)CN(C(=O)C(=O)Nc2ccccc2)CC1(C)C CC1CC(CNC(=O)CCc2cnn[nH]2)CN(C(C2C3CC4C(C3=O)C24)=O)C1 c1(SC(CC)C(=O)NCc2nnc(C(=O)O)o2)ccc(F)cc1 N1(C(CC(=O)OC)=O)CCCCC1CN(C(=O)CC1(CN(C)C)CCCCC1)C C1(C(N2C(CC(=O)NCCCn3c(C)ncc3)CCC2)=O)CC2(CC2)CO1 C1(C(N2CCCC(CCCC)C2)=O)CN(C(=O)CNC=O)CC1C1CC1 N1(C(c2c(C)cns2)=O)CC=C(C(C)(C)C(=O)N2CCCC(C)(C#N)C2)C1 c1(C(N2CC(NC(C(C)Cn3cccn3)=O)C2)=O)c(C(F)(F)F)cnn1C c1(C(=O)NC2CCN(C(C3(C)CCC(=O)C3)=O)C2)cnn2ncccc12 CCCCCC(=O)NCC(C)(CNC(C1CCN(CC)C1)=O)OC C(=O)(CCCC(=O)NOC(C)(C)C)NC1CN(C(COCCC#C)=O)CC1(C)C c1(C(N)=O)ccc2c(c1)C(C(=O)Nc1cccc3c1CN(C(N)=O)C3)CO2 Cn1cnc2sc(C(=O)NC3CC(CNC(=O)Cc4cnc[nH]4)C34CCC4)cc12 CC1c2ncc(C(=O)N(C)CCN(C)CCO)n2CCN1C(=O)Cc1cscn1 C#CCCCC(=O)NCC1(C)CCCN1C(c1cc(C)c[nH]1)=O N#Cc1cnc(C(=O)NC2CC(O)CN(C(=O)CN3CCS(=O)CC3)C2)c(Cl)c1 c1(C(N2CC(O)(CCNC(C(C=CCCC)O)=O)C2)=O)n[nH]c2ccccc12 C(=O)(C1=Cc2ccc(Cl)cc2OC1)NC(CC1CN(C(CN(CCC)C)=O)C1)C O=S(=O)(c1ccc(NCCc2ccns2)c(Br)c1)NCCCC1CCCC1 N1(C(CC2CC(OC)C2(C)C)=O)CC2CC(C1)C2NC(c1oncc1C)=O N1(C(C(C)NC(=O)OC)=O)CC(C)(C)CC1C(=O)NC(c1ncccc1F)C N1(C(C2(C#C)CCCC2)=O)CC=C(CC(=O)NC2CCCC(C(N)=O)C2)CC1 N1(C(CCCNS(C)(=O)=O)=O)CC(F)CC1CNC(=O)C(C)=CC(C)(C)C C1(C(N2CCC(C(C)NC(C3CC4C=CC3C4)=O)C2)=O)(CC)CCNC1=O C1(c2ccc(CC)cc2)CN(C(=O)CSC(C)C)CCN1C(=O)Cn1cnnn1 C1(NC(C=CC2N(C)CCC2)=O)CC2(C1)CN(C(=O)CC13CCC(CC1)CC3)C2 C=CCC(C(=O)N1CCC1CNC(C1(c2ccc(OC)cc2)CC1)=O)N(C)C CCC(C)CC(C)N(C)C(C1CC(N(C)C(c2cnncc2C)=O)C1)=O c1(-c2cn(C(C)C(=O)NCc3ccn(C(F)F)n3)nn2)c(F)cncc1F N1(C(C2(NC)CC2)=O)CC(OC)CC1C(=O)NCc1nnn(C)c1C n1(CCN(C(=O)C(O)CC2CCCC2)CC)cc(CNC(=O)C(C)O)nn1 c1(C(N(CC(C)(C)CNC(=O)CC2(C)CC2(F)Cl)C)=O)[nH]nc2ncccc12 C(=O)(C=C1SCC(=O)N1C)NC1COC2CN(C(C(C=C)(C)CCOC)=O)CC21 c1(CC(=O)NC(C)(CNC(=O)CN2CCCCC2=O)CO)cnn2c1CCCC2 C1(NC(C2(CC=C)CCN(C(C3C(C)C3C)=O)C2)=O)CCCC(O)CC1 C1(NC(C(CC)SC)=O)CN(C(c2c(F)ccc(OC)c2N)=O)CCC12CCC2 c1(CNC2CC(NC(Cc3c(OC)cc(F)cc3)=O)C2)c(Br)cc(Br)c(C)c1Br N1(C(C2(C(=O)NC)CC2)=O)CCCC(O)(CNC(=O)C(C)c2cccs2)C1 C(C(C)(C)C(N)=O)NC(C1(NC(C2C(C)CC2)=O)CC(CO)C1)=O c1(C(=O)NC2C(NC(CC(CCC)C)=O)CC2)cn(CCO)c(=O)nc1O C1(C(=O)NCCC)CN(C(=O)CN(CC)Cc2ccc(C)cc2)CCO1 C(=O)(CCCS(C)(=O)=O)NCCOCCCNC(c1c(C#C)c[nH]n1)=O c1(C(N(C)CC2OCCN(C(C(C)C(C)(F)F)=O)C2)=O)cc(S(N)(=O)=O)oc1Cl c1(C(N2CC(O)(CN(C(c3nn(CC)c(C)c3)=O)C)C2)=O)cc(OC)ccc1F C1(C)(C(=O)NC(C)CN(C)C(c2occc2C2CC2)=O)CCN(C)C1 C1(NC(C(CC)N(C)C)=O)CN(C(=O)COCC2CCC2)CCC12CCOCC2 C1(NC(C(N2CCC(C(C)(O)C(F)(F)F)CC2)=O)=O)CNc2ccccc2C1 c1(C(=O)NCCC2OCCCN(C(CC(C=C)C)=O)C2)nn(C)c2ccccc12 c1(C(=O)NC2CCC(NC(C3CCN(C)CC3)=O)CC2)ccc([N+](=O)[O-])c(Cl)c1 C(=O)(CC(C)(C)OC)NCC(CC=C)NC(C1CC(n2cnnc2)C1)=O N1(C(COCCC=C)=O)CC(NC(=O)CC(C)C)CC2(CCOCC2)C1 C1(C(C)NC(CSCC)=O)CCCN(C(c2[nH]cnc2C)=O)C1 C1(NC(c2ccnc(C(=O)O)c2)=O)C2Cc3c(Br)cccc3C12 C(=O)(C(C)CCC(C)(C)C)N1C2CCN(C2)C(C)C1=O.C1(SC)CCCCC1 c1(C(=O)NC(CNC(C(CCC)OC)=O)C(C)C)cc2c(C)cccn2n1 C1(NC(c2cccc(Cl)c2)=O)CN(C(c2cn(C(F)F)cn2)=O)CC2(CCC2)C1 C1(C(=O)NCc2n(C)cnc2)N(C(=O)CN2CCC(F)CC2)CC12CCCC2 c1(C(=O)NC2(CNC(=O)C3=CCOC3)CCC2)ccc(=O)n(CCF)n1 Cc1nc(C(=O)NC(C(C)NC(c2ncoc2C2CCC2)=O)C(C)C)c(C)s1 CC1OC2CCC1(C(=O)NCCC1(NC(=O)CCCCCN(C)C)CCC1)C2 C#CCC(CC#C)C(=O)NC1(C2CCN(C(c3c(C)cc(F)cc3C)=O)C2)CC1 N=c1ccc(C(N2CCN(C(=O)Cc3csc(C(F)(F)F)n3)CC2)=O)c[nH]1 Cc1cccc(C(=O)NCCN2CCCN(C(=O)C(C)c3cc[nH]n3)CC2)c1O C1(CNC(C(CCC)c2ccc(Cl)cc2)=O)CC2CCC1N2C(=O)CS(C)(=O)=O c1(CNC(c2nnnn2CC2CCOC2)(CC)C2CCCC2)cn(C)cn1 CC(C)CCCC(C)CNC(=O)C(C)(CO)NC(=O)CC1(O)CCCCC1 C1(OCC)CCC(N(S(=O)(=O)CCOC(C)(C)C)C)CC1 C1(NC(C(CC2CC2)OC)=O)CN(C(c2ccc(C)cc2)=O)CC2(CCC2)C1 C1(C(=O)NC(C#C)C2CC2)OCCC1NC(=O)CC=CCCCCC CC1(C)SCC=C1Cc1nc(C2CC3(CCC3)C2O)no1 c1(C(N2CCC(n3cc(CC(=O)OC)nn3)(COC)C2)=O)nccc(C)c1Br N1(CC)CC(N=c2ccnc(NCC(N3CCC(C)CC3)C)[nH]2)CC1=O CC1=C(C(=O)NC2CN(C(=O)CCc3csc(Br)c3)C2)CCCO1 n1(CCOC)nnnc1C(c1ccc(C2CC2)o1)NC(C)Cc1cnn(C)c1 c1(C(N2CC(CN(C(C=CCC)=O)C)OCC2)=O)cc2c(C)cc(Cl)cc2[nH]1 c1(C(=O)NC(CCCCNC(C(OC)OC)=O)C)c(C)[nH]c2ccc(Cl)cc12 C1(N(C(CCOC(C)C)=O)C)CCCN(C(=O)C(C)Oc2ccc(Cl)cc2)C1 c1(OC)ccc2[nH]cc(C(=O)O)c2c1.C12CCCN(C1)CC2=O C(=O)(C(C)S(N)(=O)=O)NCCC(C(=O)NC(c1ccccc1)C)OC N1(C(C(=O)OC(C)(C)C)=O)CCOC(C)(CN2CCCCC2)C1 N1(C(c2c(C)nncc2)=O)C2CCC1CC(N(C)C(C1(C)CC1(F)Cl)=O)C2 C1(NC(c2ccc(F)cc2F)COC)CS(=O)(=O)CC1C c1(C(C)NC(=O)C(CCF)NC(=O)Cc2nccn2C)ccnc(F)c1 N1(C(C(F)=C(C)C)=O)CCCC1CCCNC(=O)CCc1cn(C)nn1 c1(-c2cccc(C#C)c2)cnn2cc(C(=O)Nc3ccc(O)cn3)cnc12 c1(OC)cccc(C(CNC(=O)C(C)C2CC2)NC(c2c[nH]cc2Br)=O)c1 C1(C)(C(N(CCC)CCNC(=O)CC2CN2)=O)CCOC(C)C1.OCC c1(C(N2C(C)CC(CNC(C=CSC)=O)C2)=O)ccc(O)nc1Cl N1(C(C(CC=C)C)=O)CCCC(NC(=O)CC2(C(F)F)CC2)CC1 Cn1cnc2nc(N3CCN(C4CN(C5CC5)C4)CC3)nc(N3CC4CC4C3)c12 N1(C(CC(=O)OC)=O)CCCC1C=CC(=O)N(C)Cc1cn(C)nc1C N1(C(C=C(C)C(C)C)=O)CC2C3CCC(C2C1)N(C(C12CC(C)C1C2)=O)C3 c1(C(=O)NCC(C(C)(C)C)NC(C=COCC)=O)cc(F)ccc1O C(C(C)(C)CNC(=O)CCOC1CN(C(=O)CCn2cnc(=N)[nH]2)C1)OC CC1OC(C)CC1C(=O)NCC(O)CNC(c1snnc1C1CC1)=O c1(C(N2CC(C(C)NC(=O)CNC(N3CCCC3)=O)C2)=O)cc(C#N)no1 C1(CNC(C(c2ccccc2)OC)=O)CC(F)CN1C(C1CCC(C)C1)=O N1(CC(CC(C)C)OC)CC(C#N)N2CCC1C2 C=CC1(CC(=O)NC2CCC(CNC(C3(C)CCC(C)C3)=O)CC2)CCCCC1 N1(C(c2cccc(OC)n2)=O)CCC2(C1)CN(C(=O)CCOC(C)C)CCO2 c1(C(N2CC3CC(F)(C3)C2)=O)c[nH]c2cc(F)cc(F)c2c1=O C1(CCCNC(C2(F)C(C)C2)=O)CCCCN1C(c1cccc(C2CC2)c1)=O C1C(C2CC2)CCN1C(=O)C=C(Cl)Cl.CC1(C)CCN(C2CNC2)C1 C=CCC(C)(CC)C(=O)NC(C1CCN(C(=O)Cc2ccc(C)c(F)c2)CC1)C Cc1cccnc1C=CC(=O)NC1CC2CC(NC(C3(Cl)CC34CCC4)=O)C1C2 C1(C(=O)NC2(CSC)CC2)(CNC(C2CCCSC2)=O)CCCC1 c1(C(=O)OC)nc(C(=O)N(C)C(C2CCCO2)C)cs1 Cc1nc2cccc(Cl)c2cc1C(=O)NC(c1ccccc1Br)C(F)(F)F C1(C(=O)NC(CCNC(C(C)OCCC#C)=O)(C)C)Cc2ccccc2O1 c1(C(N2C(CN(C(=O)C=Cc3cnccn3)C)CCCC2)=O)cnc(O)cc1O Cc1cc(F)c(Cl)cc1C(=O)NC1CCN(C(=O)COCCC(C)C)C12CCC2 N1(CC(=O)NCCCN(C)C)CCC(C)(N2CCCC2)CC1 N1(C(C(CCC)NC(=O)C(C)(C)C#N)=O)CCCC(C)(F)C1 C#CCCCC(=O)NCC(C1CCN(C(C2CC2OCC)=O)CC1)C C1(C(=O)NCC(CCNC(c2occ3c2CCC3)=O)O)CCC=CCCC1 c1(C(=O)NCCC(C)Nc2nc(OCC)c(Cl)cn2)cccc2nc(O)ccc12 C1(CNC(C2CC(OC)(OC)C2)=O)CC2CCC1N2C(=O)C(n1ccc(C)n1)C CCC(C(=O)NC1(C)CC(NC(c2n[nH]c(C)c2Cl)=O)C1)C(F)(F)F Cc1cc(NC(C2(C)CCCCO2)c2nnnn2CCN(C)C)c(C)c(C)c1 C1(NC(C(CC(N)=O)O)=O)CN(C(=O)C#CC2CC2)Cc2ccnn2C1 N1(C(CP(C)(C)=O)=O)CC2(CC2)CC1CC(N1CCC(CN(C)C)C1)=O C1(CNC(C2(CCCC)CCCC2)=O)CCCCN(C(=O)CCC(C)(C)C)C1 N1(C(C(CO)OC)=O)CCC(C(=O)NC(C)Cc2ccccn2)C(O)C1 C12(NC(Cn3nc(C)c(C)c3C)=O)CCN(C(=O)CSC(F)F)CCC1C2 C(=O)(CCCCCCNC(=O)C(F)C(C)C)NC(CC(=O)OCC)C c1(C(N(C2CCN(C(=O)CCOC)C2)CCC)=O)cc2c(cc1Cl)NC(=O)C2 C12(C(=O)NC3CNCC3c3cc(F)cc(F)c3)CCCCC1CC(F)(F)C2 C(=O)(C1CC(=O)Nc2ccccc21)NCC1(C(N)=O)CN(C(C=C(C)C2CC2)=O)C1 C(=O)(C(C)(C)CC(F)F)NC(CC)CCC(=O)NC(CO)CC(F)(F)F C1(CN(C(C(C)OCC2CC2)=O)C)COCCN1C(c1cc(C(C)(C)C)on1)=O n1(CC(=O)N(CCNC(C2C(Cl)(Cl)C23CC3)=O)C2CC2)nc2n(c1=O)CCCC2 c1(C(=O)NCC(CO)NC(c2nn(C)c(O)c2)=O)ccnc(F)c1N C12(C(=O)NC(C3CCN(C(c4c(C)csc4)=O)C3)C)CC(CN1C1CC1)C2 c1(OC)cncc(C(N2CC(O)(CN(C(=O)CC3CCN(C)C3=O)C)C2)=O)c1 n1(CC)c(C(=O)N(CC(C)C(=O)N2CC(F)(C(=O)OC)C2)C)cnc1O c1(N2CCC(N(C(CCC(=O)NCC=C)=O)C)C2)nc(C)cc(C)c1C#N c1(C(=O)NCCCN(C(c2ccncc2C(F)F)=O)CC)cncnc1C1CC1 c1(C(=O)NC(C2CCCC2)CNC(CC2(C)CCCO2)=O)cc(F)cc(Cl)c1O c1(C(=O)OC)cc(C)c(NC(c2nnn(-c3ccccc3F)c2C)=O)c(Br)c1 CC1(C)CCOC1C(=O)NCCn1cnc(C(=O)NCCc2ccon2)c1 c1(C(=O)NC2(C(N3CC4CCCC34)=O)CCSC2)cc(O)cc(=O)o1 C=CC(C)(C)CC(=O)N1CCN(C(c2cncc(Cl)c2Cl)=O)C(COC)C1 C(c1ccc(C#N)cc1)=CC(=O)NC1(CNC(C(N2CC(C)C2)C)=O)CCC1 c1(C(=O)NC2CN(C(C3CC(CC(F)(F)F)C3)=O)C2)ccn(CCO)c(=O)c1 c1(CN2CC(NC(c3c(C)ccnc3)=O)C(O)C2)cccc(C)c1O Cc1cc(C(=O)NCCOC2CN(C(C3CCC=CCC3)=O)C2)cc(=O)n1C N1(C(CCCC)=O)CCN(C)C(CNC(c2ccc(C3CC3)cc2OC)=O)C1 C12(NC(C(C)OC)=O)CCCC1CN(C(c1cc(C(F)(F)F)no1)=O)C2 C1(CC)CCCCC1C(=O)NCCCNC(c1cc(C)ns1)=O C1(NC(c2c(CC)cccn2)=O)CC(F)(F)CC1NC(c1ccc(O)c(Cl)n1)=O c1(OCC)ccccc1CCC(N1CC2CC2(NC(=O)CCS(C)=O)C1)=O N1(c2c(C)c(NCCC(C)CO)ncn2)CCc2cncnc2C1 C1(C(N(C2CCN(C(c3cccc(C(N)=O)c3)=O)C2)CCC)=O)OCCC1(C)C c1(OC)cncc(C(=O)NCC(O)C(=O)N(CC(O)C2CC2)C)c1 N1(C(C(C)(CO)OC)=O)CCC(F)(F)C(CNC(=O)CCCC(=O)NC(C)C)C1 N1(C(C2(CCC=C)CC2)=O)CCC(c2n[nH]cc2CNC(=O)CC(C)C)C1 c1(OC)cc(CC(=O)NC2CN(C)C2)cc(F)c1.N12CCN(CC1)C(=O)C21CC1 C(=O)(C1=CCC(C)(C)CC1)NCC(CNC(C(c1cccc(OC)c1)OC)=O)C N1(C(COC)=O)CC2CC(C1)CN(C(c1ccc(NC3CC3)nc1)=O)C2 N1(C(C(C=C)O)=O)CC2CC1CC2CNC(c1n[nH]c(C(C)C)c1Br)=O C(C(F)(F)CC(O)CO)N(C(=O)C(O)C1(NC(C)(C)C)CCC1)C C1(OC)(CO)CCN(C(c2cc(C(F)F)on2)C(=O)NCCCC2CC2)C1 N1(C(C2CC(C(=O)OC)C2)=O)CC(NC(C2CCCC(C)(C)O2)=O)C2(CCC2)C1 CCCN=C(NCc1cc(-c2ccccc2)on1)NC(c1ncccc1F)C c1(C(=O)OC)cc(C(=O)NCC2(N(C)C)CC2)n(C)n1.C12CN(CC1OC)C2=O C1(NC(c2cc(OC)ncc2)=O)CC(F)CN(C(=O)C(c2ccnn2C)C)C1 CC1=C(C(=O)N2CCC(C)C(NC(C3(C4CC4)CCC3)=O)C2)CCCO1 c1(C(=O)NC(c2ccncn2)C)coc(CNC(c2nnsc2N)=O)c1 CCCCC(C)C(=O)N1CCCC(NC(=O)Cc2csc(C3CC3)n2)C1C c1(CC(=O)OC(C(=O)OC)C)cccc(C2CC2)c1.C1C(O)CNCN1 CN=c1[nH]nc(CC(N2CC(CCNC(=O)COc3cn[nH]c3)C2)=O)s1 c1(C(N2CCN(C(c3cnc(Cl)s3)=O)CC2C2CC2)=O)ccnc2[nH]ncc12 CN1CC(NC23CNC(C)(C2)C3)CC12CCC2 c1(C(N2CCC(N(C(=O)CC34COCC(C3)C4)C)C2)=O)ccc2[nH]c(=N)sc2c1 O=C(C1=CS(=O)CCC1)NCC1COCC1NC(=O)CSc1ccccc1Cl C1(C(N(CC(=O)NCCC(F)(F)Cl)CCOC)=O)C2(CC2)C12CC2 c1(CNC(C23CC(CO)(C2)OC3)=O)cccc(NC(=O)C(c2ccccc2)O)c1 C(=O)(C(C)(C)C(C)OC(C)(C)C)N1CCC(OCCNC(C=CCOC)=O)CC1 N1(C(c2c(C)cc(C)o2)=O)CC(C(=O)NCC2(O)CCC(C)(C)C2)CC(C)(C)C1 c1(C(=O)NCC2N(C(C(F)OC)=O)CC2)cnc2ccccc2n1 C(=O)(C(C)(C)CC(=O)N(C1CCN(C(C2CN(CC(C)C)C2)=O)CC1C)C)OC c1(N2CCC(C)C(NC(C(N3CCOCC3)C)=O)C2C)nc2ccc(F)cc2o1 CCC(CCOC)C(=O)NCC1CCCN1C(C1CCC(C)C1)=O C1(C(N(C2CCN(C(c3coc(C)c3)=O)C2)CC(=O)OC)=O)CCCCC1 c1(C(N(CCOCCCN(C(C2C=C(C)CS2)=O)C)C)=O)ccc(F)cc1F N1(C(c2nc(CNC(C3(OCC)CC3)=O)oc2)=O)CCC2CCC12 C1(CNC(c2cncc(C(F)(F)F)c2)=O)CN(C(c2ccccc2Cl)=O)C2CC12 c1(CNC(C(=O)NCc2nc(-c3ccc(C)o3)sc2)=O)cccc(C2CCC2)c1 C(=O)(C(CCC(C)C)NC(C)=O)N1CC(C)(N(C(C(F)=CCC)=O)CC)C1 C12(C(N3CCCC(C(=O)NC(C(=O)NCC)(C)C)C3)=O)CCC(CC1)CO2 N1(C(C2N(C)CCN(C(C3CC(OC4CC4)C3)=O)C2)=O)CCC12CCCCC2 c1(C(N2CCC(Cc3ccccc3)C2)C(=O)NCCCF)ccc(F)c(SC)c1 c1(C(=O)NC(CNC(C2CC(C)(C(=O)OC)C2)=O)(C)C)ccc(Br)cc1 C1(C(N2CC(C)C(F)(F)C2)=O)CC(O)C(O)CC1CNC(C1CC(=O)N(C)C1)=O C1(CC(=O)N(C2CC2C2CC2)C)CN(C(C2(F)CC=CCC2)=O)CCO1 C1(C(=O)NCC(=O)N(C)C)C2C(CN1Cc1c(F)ccc(F)c1O)C2(C)C C1(NC(c2cc(C)[nH]n2)=O)CC2CCC1CN2C(=O)CC1(C)CCOCC1 Cc1cc(C(N2CC(NC(=O)C(C)Oc3ccc(O)cc3)C(C)C2)=O)ncc1F C1(N(C(CCNC(C)=O)=O)C)CCN(N(C)C2CC3(CC3)C2)CC1 CC(CC1CCCCC1)C(=O)NCCN(C(c1coc(Cl)n1)=O)C1CC1 c1(C(=O)NC2C(NC(CNC(CCC)=O)=O)CS(=O)(=O)C2)n[nH]c2ccccc12 CCC(CC(F)(F)F)C(=O)Oc1ccc(OC(F)(F)F)cc1C(=O)OC(C)(C)C Cc1sc(C(=O)NCCCCC2CCCN(C(C3C(C#N)C3(C)C)=O)C2)nc1O c1(C(=O)Nc2ccc(C(=O)NC(C)CC(=O)O)cc2)cc2c(nn1)CCOC2 CC1(CNC(=O)C2=CSCCO2)CCN(C(c2cc(C3CCC3)on2)=O)CC1 C(C(=O)N1CCC(C(=O)N(C)Cc2cocn2)C1)(C(C)C)NC(C)=O c1(C(N(C2CCN(C(c3cccnc3)=O)C2)C)=O)c(F)ccc(F)c1Cl CCC(CC)C(C(=O)N(CCC(=O)NCC1OCCC1(C)C)OC)OC Nc1c(C(=O)NCCNC(c2cnc(O)s2)=O)sc2nccnc12 C12CCCCN(C1)C(=O)CCCn1cc2nn1.C1(COC)CS(=O)(=O)CCO1 C1(CCNC(C2(OCC)CCC2)=O)C(C)CCCN1C(=O)CN(C)C c1(OC)ccnc(C2(C(N3CC(CCNC(C4(F)CCOC4)=O)C3)=O)CCC2)c1 N1(C(C(N2CCCC3=NC=C3C2)=O)=O)C2CCC1C1CNCC21 c1(C(=O)NC(c2ccccc2)(COC)C)cccc2cc(Br)cnc12 N1(C(C(COC)OC)=O)CCCC(n2cc(C3CCC(OC)CC3)nn2)C1 N1(C(C(CCC)O)=O)CC2(CCC2)CCC1CNC(C1CC2(CCC2O)C1)=O N1(C(CCC2CCCN(C)C2)=O)CCCC2CN(C(=O)CS(=O)(=O)C3CC3)CC12 CCC(C(=O)NCc1cn(CC(=O)N(CC)Cc2cncn2C)nn1)SC CCCC(C(O)C(=O)NCCC(O)C(F)F)NC(=O)CCC(C)(C)C C1(C(N(C(CCNC(C2C(=C)C2)=O)C)C)=O)C2CCC1(c1ccc(F)cc1)C2 C(CCCCCCCO)N.C(=O)(C=CS)OC C1(C(N(CC=C)CCO)=O)CN(C(=O)CCC2CCCN2C)CC12CC2 c1(C(=O)NC23CC(NC(CCC4CCC(C)O4)=O)(C2)C3)ccc2c(c1)CCO2 c1(C(=O)OCC)ccc(CN2CCC(O)C2C(=O)Nc2cc(CC)n(C)n2)nc1 CC1(C)CC(NC(=O)CCc2cnco2)CN(C(c2ncoc2C2CC2)=O)C1 N1(CCN(C2CCCC2O)C(C)=O)CCCC2(C1)CN(C)C(=O)O2 N1(CC)CC2CC1CN2C(=O)C(C1(C)CC1)NC(=O)CC(C)(C)CC C1(NC(CNC(C(C)C)=O)=O)C2CCCN(C(=O)OC(C)(C)C)C2C1(C)C Cc1c(C(=O)NC2(CNC(c3cccc(=S)n3O)=O)CCC2)cnc2ccnn12 N1(C(C23C(C(N)=O)(CCC2)C3)=O)CC2(CCN2C(c2snnc2C2CC2)=O)C1 c1(C(N(C)Cc2c(C)cncc2)=O)cc2c(c(S(N)(=O)=O)c1)OCC2 CCC(CCCC(=O)N1CCCC1CN(C)CC1CCCC1)NC(=O)CCSC c1(C(N2CC(NC(C(C3CCC3)OC)=O)C(O)C2)=O)cc(C)cc(C)c1N C1(C)(C(=O)NCCCC#C)CCCN1C(c1cccnc1C(F)(F)F)=O c1(CC(=O)N(C(CNC(C2(CCC=C)CC2)=O)C)C)conc1C C#Cc1cnn(CC(N2CCC(C)C2C(=O)NCCCCC(C)C)=O)c1 C1(C(=O)NC2CC(CNC(c3ccc(C(C)(C)C)s3)=O)C2)C2CC2C2CC12 c1(C(=O)NC2CCC(N(C(CC(=C)Br)=O)C)C2)cc(N)c(F)cc1F N1(C(c2ccccc2)C)CC(CNC(=O)C(F)(F)Sc2cnn(C)c2)CC(F)C1 c1(C(=O)NC(C)CCCNC(C2CCCSS2)=O)ccc(-n2ccnc2)cc1 CCC(CNC(C1CCCCC1OC)=O)(CC)NC(c1ccc(OC)nc1)=O C(=O)(CC(=O)NCCCCNC(C1CCCN1c1cnccn1)=O)N(C)C c1(OC)cc(C(F)F)c(C(N2CC3CC3(CNC(=O)C(O)C3CCC3)C2)=O)cn1 C1(C(N(OC)CC2CCCCC2)=O)CCCCN(C(C2CC(C)C2)=O)C1 c1(OC)ccc(Cl)c(NC(=O)CN2CCC(OC3(C)CCS(=O)(=O)C3)CC2)c1Cl N12CC3(CCC1CC3)NC2=O.N1(c2c(C)ccc(CO)c2)CCOCC2(CC2)C1 C1(C(N2C(CNC(c3nnc(C)s3)=O)CC(OC)C2)=O)CCc2ncc(C)n2C1 C(=O)(C1=C(C)CCC1)N1CCC(c2ccccc2)(NC(C=CC(CC)C)=O)C1 Cc1ccc(S(=O)(=O)N2CCN(C(=O)Cc3ccc(S(N)(=O)=O)s3)CC2)cc1 CC(CN1CCOCC1)C(=O)NCC1CC(NC(C2CC=CCO2)=O)C1 C1(C(=O)NCC23CC2CN(C(=O)CC2=CCOCC2)C3)CCc2[nH]nc(O)c2C1 c1(NC2C(C)CN(C(c3coc(Br)n3)=O)CC2)ncc(Br)cc1C#N CCC(CC)CC(=O)N(CCC(C)(C)NC(=O)C=Cc1cccn1C)C N1(C(CC(C=C)C)=O)CCC2C(NC(C3CCCC3C3CC3)=O)C2C1 N1(C(C2(C(CC)(F)F)CC2)=O)CC(CNC(=O)Cn2nnnc2C)(OC)C1 C=CCC(CC)C(=O)NC(CC)CCC(=O)NCC(O)C(N)=O C(=O)(CCCC(=O)N1CCN(C(=O)Cc2ccc(C)c(Cl)c2)C2CC12)NCCC N1(C(C(c2cc(F)cc(F)c2)C)=O)CC2CN(C(C3CCCS3(=O)=O)=O)CC2C1 C1(C(=O)NC(C)C(C)(C)NC(c2cn3ccnc3cn2)=O)CC2CSCC(C1)C2 c1(OC)cc(C2(C(=O)N(CCC(=O)O)C)CCC2)ccc1Br N1(C(c2c(C)cc(C)[nH]2)=O)CCCC2(NC(c3cc4cc(Cl)sc4[nH]3)=O)CC2C1 C1(C)(CNC(c2cc(CC)nc(O)c2)=O)CN(C(=O)CCNC(C)=O)C(C)(C)C1 C1(CNC(c2c(C)ocn2)=O)CC2COCC2N1C(=O)CC(C)C(F)(F)F C1(N(C(C=CC=CC)=O)C)CCCC2CN(C(c3ccc4cncn4c3)=O)CC12 c1(NC(C2N(Cc3c(F)cc(C)cc3Br)CC2)=O)ncc(I)cc1[N+](=O)[O-] C1(C(=O)NC2CCCN(C(C(C)NC(C)=O)=O)CC2)CCc2nnc(O)cc2C1 C1(C)(CNC(C(CC2CCC2)OC)=O)CCC(NC(=O)Cc2ccoc2C)C1 Cc1cc(C(=O)NCC2(O)CC(NC(c3ccc(O)cn3)=O)C2)nn1C(C)C N1(C(C(COC)(F)F)=O)CC2OCC(NC(=O)CN3CCC(C)C3)C2C1 C1(C(=O)NCC2CC(CN)C2)CCCN1C(C1(O)CC1)=O.c1(C=O)cccs1 c1(C(=O)NC2C(C)N(C(c3ccsn3)=O)CCC2)[nH]c2ccccc2c1Cl C12(C(N(C3CCCC3)CCNC(c3ncc(F)cn3)=O)=O)CCCCC1C2(F)F c1(CC)[nH]nc(C(=O)NCc2cn(CCNC(C3CN(C(N)=O)C3)=O)nn2)c1Cl N1(C(C2(C#N)CC(C)C2)=O)CC(C2CCCN(C(C3(n4cncn4)CC3)=O)C2)C1 C1(C(=O)NCC(=C)CC)CCC(O)CN1C(c1ccc(OC)s1)=O c1(CN(C(=O)Cn2nnc(CN(CC(=O)OCC)C)n2)CC)cccc(Cl)c1 n12cc(nn1)CC(=O)N(CC)CCC2.n1(CC2(CC)COC2)cc(C(=O)O)cn1 C1(CNC(c2cc(C(=O)OC)no2)=O)CCCCN(C(=O)CC2=CCCC2)CC1 CCC(CC(F)(F)F)NC(C1(CC)CCCN1C(=O)CCc1ccco1)=O C1(C(=O)NC2(CC)CN(C(C3CCCN3C)=O)C2)CCS(=O)(=O)C1 CC1CC(C(=O)NC23CC(C2)N(C(C2CCCOC2)=O)C3)CC(C)O1 CCC(C)C(C(=O)N(C(C)C(=O)NC1CNC(=O)OC1)C1CC1)N(C)C c1(OC)noc(C)c1C(=O)N(CCCCN(C(=O)CCc1ccc(=N)[nH]c1)C)C C1(OC)CC(CNC(c2ncccc2C)=O)N(C(=O)C(N2C(=O)CCC2=O)C)C1 c1(C(C(=O)NCC)N(C2CNC(=O)C23CC3)C)c(C)cccc1C C(=O)(C1=NOC(C)(C)C1)NC1CN(C(C=C(COC)C)=O)C1 N1(C(c2c(C)n[nH]c2)=O)CC2CN(Cc3ccc(CC(=O)O)cc3)C2C1 C1(CNC(c2snc(O)c2Cl)=O)CN(C(C2(F)CC2)=O)C2CC12 C1(C(=O)NCCN(C(C(=O)N(C)C)=O)C)CC12CCS(=O)(=O)CC2 c1(C(=O)NC2C(C)N(C(=O)CC3CC3)CCC2)ccc2c(c1)C(C)(C)C(=O)N2 c1(C(N2CC(O)CC2CO)=O)cc2c(-c3ccc(O)c(F)c3F)cccc2s1 N1(C(CCC(C)(C)NC(c2c(Cl)cn(C)n2)=O)=O)CCC2(CCCO2)CC1 CCCC(CCCNC(c1ccc(Cl)cn1)=O)Nc1ncnc(Cl)c1C c1(C(N2CCC(NC(C(CC)=O)=O)C(C)(C)C2)=O)ccc2sccc2c1O C(=O)(C1CCCn2nccc21)N1CC(F)CC(NC(c2c(=O)ccn(C)c2)=O)C1 C(=O)(CN=c1[nH]c(C)cs1)N1CCC2CN(C(CCc3nc(C)sc3)=O)CC21 C1(NC(CC(CC)N(C(=O)C=Cc2cocn2)C)=O)CCCCCC1F C(=O)(CCC(=O)N(CCC(C)NC(C1CCCCS1)=O)C)Nc1nnc(CC)s1 CC1CN(C(=O)CCc2cccnc2Cl)CC1NC(=O)C(C)c1ccsc1 C1(C(N(CCCC)C(C)C)=O)CN(C(c2sccc2C)=O)CCC1O N1(C(COCCCCC)=O)CC2(CNC(C3CC34CCSCC4)=O)CCC1CC2 C1(C(C)NC(C2(C3CCCO3)CCC2)=O)CCCN1C(=O)CNS(=O)(=O)C1CC1 N1(C(c2cc(C)no2)=O)CCC(C2CC2)(CNC(c2ccc(O)nc2)=O)C1 CCCC(C(=O)NC1CCN(C(=O)Cc2nc(C3CC3)cs2)CC1C)C(C)C C1(OC)CC(C(=O)NCCN2CC3CC3C2)N(C(C2C=CC=CC=C2)=O)C1 N1(C(C(=O)CSCO)=O)CC2COCC(C1)C2CC(=O)NCC#N.C=CCN C(=O)(C(O)C(F)(F)F)N1CCN(C(C(C)Oc2cccc(Cl)c2)=O)CC1 CCC(CC(=O)NC1CN(C(=O)Cc2nn(C)cc2Cl)CC1n1ccnn1)OC c1(C(=O)NC2CC(CCNC(C3N(C)CCC3)=O)C2)ccc(C(F)(F)F)c(F)c1 c1(C(=O)NCC2N(C(C(C=CCCC)O)=O)CCOC2)[nH]nc2ncccc12 C1(CNC(C(CC=CC)C)=O)CN(C(c2cnn(CCC)c2)=O)CCCO1 c1(C(=O)NCC(C)N(C)C(c2cc(Br)no2)=O)cccc(F)c1C#N C12(C(=O)NCC3CCC(NC(C4C(CC)C4)=O)CC3)CC(C1)S(=O)(=O)C2 C(CC(C)(C)C)(C(=O)N1CC(O)(C(F)(F)F)C1)NC(C(C)OC(C)=O)=O C(=O)(C1=CC2(CCOC2)C1)N1CC(CCNC(C(CC(C)C)(F)F)=O)OCCC1 N1(C(CNC(CCC)=O)=O)CCCN(C(C2CCN(C=O)O2)=O)CC1.C(C)(C)(C)O C1(N(C(C(CC)N(CC)CC)=O)C)CCCCC1NC(C12CC(C(C)C)(C1)C2)=O C1(NC(COCCCOC)=O)CC(O)CN(C(=O)CN2CCCNC2=O)C1 c1(C(=O)NCC(CC)(C)NC(=O)CCc2csc(C)n2)cnn2ncccc12 C1(CC(=O)N(C2CC(NC(C3CCN(C)C3)=O)C2)C)CCC(C)(C)O1 c1(OCC)oc(C)nc1C(=O)NCC1CCC(F)(CNC(C2(COC)CC2)=O)C1 c1(N2CCC(N(c3snc(CC(=O)OC)n3)C(C)=O)C2)ncc(OC)cn1 C1(CC(=O)NCC(CNC(c2cnn[nH]2)=O)OC)CC2CCC1CC2 C#CCC(C)(C)C(=O)NC1CCCC(CNC(c2occc2F)=O)C1 C(c1cc(Cl)ccc1Cl)=CC(N1C(CNC(c2n[nH]c3c2COC3)=O)CCC1)=O C(CC(C)C)(C(=O)NCC1(C(N)=O)CN(C(c2cc(C#N)c[nH]2)=O)C1)NC(C)=O C(=O)(C(C(C)C)N(C)C)NCC1(OCC)CN(C(=O)C(F)C(C)C)C1 c1(CC)ccc(-c2ccnc(CC(=O)NCCc3c[nH]nc3C)c2)cc1 C1(NC(Cc2ccc(C(C)=O)s2)=O)CCCCN(C(c2c(C)coc2C)=O)C1 CC1CCCC=C1C(=O)NCC(CC(=O)NCC1CCC(=O)N1)C1CCC1 N1(C(C(COC)C)=O)CC(NC(=O)C(C)(C)C)CCC(O)C1 c1(C(=O)NC(CNC(C(CC)(C)CO)=O)C)[nH]c(C)c(S(N)(=O)=O)c1C c1(C(C)C)cccc(C(C)(C)CN2CCC(Cc3ccc(Cl)cc3)C2)n1 C1(NC(C=CCN(C(=O)C=Cc2cocn2)C)=O)CC1C1CCOCC1 Cc1ccc(CS(=O)(=O)NCCC2CC(F)C2)cc1F N1(C(C2C(=C)C2)=O)CCC(F)C(NC(=O)CCc2nc(CCC)no2)C1 C1(CNC(c2ccc(CCC)s2)=O)(NC(=O)Cc2cccn2C)CCCCCC1 c1(CN(C(CNC(CNC(C(C=CC)O)=O)=O)=O)C)ccc(C)nc1 c1(COCC(=O)NC(C)(C)CCNC(=O)CC2(C)CC2F)ccc(F)cc1 C(CCC(C(=O)NCCCSC(F)F)NC(=O)Cn1cnnn1)OC n1(CC)nc(C)c(NC(=O)CC(C)CNC(=O)Cc2ccn(C)c2)c1C c1(CCNC(N2CCC(CCNC(=O)OC(C)(C)C)C2)=O)ccc(F)cc1O c1(CC2C(N)CN(C(=O)C(N3C4CCC3CC4)=O)C2)cnc2ccccc2n1 c1(C(C)NC(C(CC)N(C(c2c(CCC)nco2)=O)C)=O)cnccc1C C1(CC)CN(C(c2conc2CNC(=O)C(C)n2cccc2)=O)CCN1C C1(C(N2C(CCNC(C#CC3(C)CC3)=O)CC(F)(F)C2)=O)CCC(=C(F)F)CC1 CCC(C)CC(C(=O)N(C)CCC1CCCC1)NC(=O)CCOCC C12(C(N3CC(C#CC)C3)=O)CCCC1CCN2C(c1csnc1C)=O N1(C(c2c(C)cc(F)cc2)=O)CCC2(CC1)CN(C(=O)CSC1CC1)CC(C)O2 CC1(CNC(C2(F)CCCC2)=O)CC(NC(=O)CSCC2CCCO2)C1 c1(C(N2CC3CN(C(Cn4c(C)nnn4)=O)CC3C2)=O)cccc([N+](=O)[O-])c1Cl c1(NC(C2C(C)=CCC=C2)=O)ccc(NC(c2ccc(O)cc2F)=O)cc1F C#CC1(C(=O)NCCc2cnc(C)o2)CN(C(=O)C(c2ccn(C)c2)C)C1 C(=O)(C(F)(F)C(F)(F)C(F)F)NC1CCC(CNC(=O)C2=C(Cl)CCC2)C1 O=C(CCCCCCCO)NCCCN1CCOCC1 C1(C(N2C(C)CC(NC(c3cc(CC)nn3C)=O)C2)=O)CCc2cncn2C1 c1(OC)cc(C)ccc1C(=O)NC1CCCN(C(=O)CC2CCC(C)C2)C1CO N1(C(C=CC=CCC)=O)CC=CC1C(=O)NCCCCCC C1(CC)CN(C(=O)C(C)(O)c2ccccc2)CCN1C(c1ccc(Br)o1)=O C1(COC)(NC(=O)C2CC2)CCN(C(C)=O)C1 N1(C(c2nc(C(C)(C)C)sc2)=O)CC2(CCC2NC(=O)CNS(N)(=O)=O)C1 N1(C(CCC#C)=O)CCCC(O)(CNC(=O)C(CC)NC(=O)CC)C1 c1(CC(N2CCN(C(c3cc(F)cnc3Cl)=O)C3CC23)=O)cc(O)cc(Br)c1 C(CN=c1[nH]c2c(c(=NC(C)CC3CCCCC3)[nH]1)CSC2)n1c(C)ncc1 c1(OC(C2(OC)CCSC2)=O)cccc(C2CC2)n1 C(CC(C)(C)C(c1nnnn1CCOCCO)NC1(CSC)CC1)OC.C1CC1 N1(C(C=CC(C)C)=O)C2CCC1C(CO)N(C(=O)CC1CCCN1C)C2 CC1(C)CC(CNC(=O)CC(F)(F)Cl)CN1C(=O)Cn1cccc1 C12(NC(C3C(=C)CC3)=O)CC(NC(=O)Cc3cn(Cc4ccccc4)cn3)(C1)C2 C(=O)(C1=CC2CCCCCC12)NCC(C)NC(C1(c2nccs2)CCC1)=O Cc1cc(C(=O)N(CCCCNC(=O)CN2CCC(C(N)=O)CC2)C)c(C)cn1 C1(CNC(=NCCC)NCCCN2CCN(C)C(=O)C2)Cc2ccccc2C1 N1(CC2C3(CCN(C(=O)OC(C)(C)C)C3)C2)CCc2cccc(Cl)c2C1 O=C(CC(F)(F)C(F)F)N1CC2(C(=O)NCC3(CF)CC3)CC1CCO2 C12CCCN(C1)CC(=O)NCC2.c1(CC)cc(NC(=O)Cc2cnc[nH]2)n[nH]1 c1(C2(NC(C(C(C)OC)O)=O)CC2)cccc(C)c1F c1(N(CC(C(C)C)C)C)ccc(S(=O)(=O)NC2COc3ccc(Br)cc32)cc1F C1(C(N(C2CCCCC2)CC)=O)CCCN1C(c1sccc1CO)=O Cc1ccc(CC(=O)NCC2=CCN(C(c3ccc(Cl)cc3)C)CC2)c(Cl)n1 C12(NC(=O)CCc3ccc(Cl)c(F)c3)CCCC1CN(C(c1ccon1)=O)C2 O=S(=O)(c1cncc(Br)c1)N1CCC12CN(Cc1nccnc1Cl)C2 c1(C(=O)NCC(C)(C2CC2)NC(CCCCCC=C)=O)cn2cccc(Br)c2n1 c1(C(N2C(CNC(c3cn(C)c(=O)cn3)=O)CC2)=O)nccn2c(Br)cnc12 N1(C(c2ccc(F)c(OC)c2F)=O)CC2CCCC(C1)N2c1ncccc1C#N c1(C(=O)NCC(CNC(Cc2ccc(CC)cc2)=O)CO)c(C)ccnc1O C(=O)(C(O)CC(F)(F)F)ONC(C1N(C(c2c(C)cc(F)cc2)=O)CC=C1)=O Cc1c(C(=O)NCC2CCCN(C(=O)Cc3cc(Cl)cs3)C2)ncn1C C12(C(=O)NCc3cc(C(=O)NC(c4n(C)ncc4)CO)sc3)CCCC1CCC2 c1(C(N(C2CCC(NC(C(C)NC(COC)=O)=O)C2)C)=O)cnc(OC)nc1 n1(CC)nc(C)c2cc(C(=O)NCC3(F)CC(NC(=O)C=C(Cl)Cl)C3)sc12 C1(C(=O)Nc2cc(C)cc(C)c2)CC2CC1CN(C(=O)Cn1nc(C)cc1C)C2 c1(OC)cccc2c1CCC2(CO)NC(=O)NCC(N1CCOCC2(COC2)C1)=O c1(CC)ncncc1C(=O)N(CC(C)NC(=O)Cn1cccn1)C C1(C(N2CC(NC(c3nc(-c4ccc(Cl)cc4)ns3)=O)C2)=O)CC(C2CCCC2)C1 Cn1cc(CNC(=O)CCCC(C)(C)O)c(O)nc1=O C(=O)(C#CC1CCOC1)NC(CCC(=O)NCC1(OC)CCCCC1)(C)C N1(C(C2CCC(CC)CC2)=O)CC2OCCN(C(=O)Cc3cn(C)nc3Cl)C2C1 C1(NC(c2c(C)coc2)=O)CN(C(c2n[nH]cc2Cl)=O)C2CCCCC12 C(=O)(CC(CN(C)C)CC)N(C(C)C(=O)N1CCC1)CC=C.C1CC(=O)N1 CC1CN(C(=O)Cc2ccn(C(F)F)n2)C(C)CN1C(=O)CSc1nnc(S)s1 N1(C(C2(NC(CC(C)OC)=O)CC(O)C2)=O)CCC(CC(C)O)CC1 Cc1nc2c(s1)CN(C(C1CC(F)CN1C(=O)CCCC(F)(F)F)=O)CC2 c1(N2CCC(C(=O)NOC3CCCNC3)C2=O)cc(F)cc(F)c1 c1(C(C)=O)c[nH]c(C(=O)N(CCC(=O)NCC(=O)N(C)O)C2CC2)c1 C1(COCCC(=O)O)CCN(C(=O)CCc2ccc[nH]2)CC1 n1(CCC(=O)NC2CC(C)N(CCc3cnccn3)CC2)cnc2ccccc12 C(c1nnc(C(C)C)o1)=CC(=O)N(C)CC1CN(C(C(CC)C)=O)C1 c1(C(N(C)CCNC(=O)CSCC(N)=O)=O)nc2n(c1Br)CCC2 C(=O)(C1c2ccccc2C2CC1C2)C(=O)OCS(=O)(=O)CC1(NC(C)(C)C)CCOC1 C1(N(CC(C)O)C(c2cccn2C)=O)CC12CCNCC2 Cc1cc(C#N)ccc1-c1nc(C)c(NC(c2cccnc2O)=O)s1 O=CN1CCCC1C(=O)NCCC(=O)NCC(O)C(F)(F)F CCN=C(NCC1OC(=O)CC1(C)C)N1CCN(C(c2cccc(F)c2)C)CC1 C1(CNC(C=NOC)=O)CCCC2(CN(C(=O)C(=O)CC(C)C)C2)O1 c1(OC)ccc2ccccc2c1CN1CCCC1C(=O)Nc1ccc(C)nc1Cl N1(C(C=C(CC)C)=O)CCOCC1CNC(=O)CN(C)Cc1ccc(Cl)s1 c1(C(N2CC(CC)C(NC(C3CCC(F)(F)C3)=O)CC2)=O)cnc2[nH]ccc2n1 C(=O)(C#CC1(C)CCCO1)N(C1CCN(C(c2nncs2)=O)CC1)CC c1(C(N2CC(CNC(C(C)C3CC3)=O)C(C)C2)=O)cccc(F)c1Br C1(NC(c2coc(C(F)(F)F)c2)=O)CCN(C(C2(C3CCCO3)CCC2)=O)CC1 C(=O)(C(O)CC(F)(F)F)NC(CC(=C)C)C(=O)NC1(C)CCSC1 CC(C)CC(C)(O)C(=O)NCC1(F)CCC(NC(=O)CCC(C)(C)F)C1 C(=O)(CCCCC#N)NC1(C(F)F)CC(NC(C2OCCC(C)C2)=O)C1 c1(OC)ncc(Cl)cc1C(N1C(C(N2CCCC(N(C)C)C2)=O)CC2CC12)=O c1(C(N(C2CCN(C(=O)CC3CC4CC4C3)C2)C)=O)nn(C(F)F)cc1Cl C=CCC(CNC(C12CSCC1C2)=O)C(=O)NC1(CCO)CCCCC1 C1(C(=O)NC(CC=C)C(=O)NCCOc2ccccn2)CCC(O)CN1C c1(CC)c(OC)cccc1C(N1CCC(F)(CNC(C2(CF)CCC2)=O)C1)=O CCC(CC(=O)NCC1CC(C)CO1)OC.C12CCN1C2=O C1(CNC(CNC(=O)OC)=O)CCCCN1C(=O)Cn1ncccc1=O C(=O)(CCCC(=O)N1CC(NC(=O)C=Cc2cncs2)C2CC12)N(CC)CC C1(NC(CCC(N)=O)=O)CC2CC(NC(c3cnc(O)c(Br)c3)=O)C2C1 CCCCCCCC(=O)N1CCCC(CNC(=O)C(N2CCN(C)CC2)C)C1 Cc1cc(F)cc(C)c1C(=O)NC(C)CN(C)C(c1cc(O)cc(=O)o1)=O C(C)(CCC(=O)N(C1CCCN(C(c2ccoc2Cl)=O)C1)CC1CC1)OCC C1(NC(c2c(CC)non2)=O)CN(C(=O)Cc2nc(=N)[nH][nH]2)C2CC12 C(=O)(CC(C(=O)N1CC(NC(c2ccoc2)=O)CC(C)C1)c1ccccc1)OC C1(CNC(COCC)=O)CN(C(c2ccc(SCC)s2)=O)CCC12CCOCC2 c1(C(=O)NCCCN(C(=O)CN2CCC2)C(C)C)c[nH]c(C(F)(F)F)c1 c1(C(N2C(CNC(CCCCC=CC)=O)COCC2)=O)cnc(N)c([N+](=O)[O-])c1 CC1CCCN(C(C2CN(C(=O)C(N)=O)CC2C)=O)C1CO c1(C(=O)NC(CN(C)C)C(N2CCC(CC3CC3)CC2)=O)ccc(CO)cc1 c1(CSCC(=O)N(CC(C)NC(C2(F)CC=CC2)=O)CC)ccccc1Cl C1(CNC(=O)CCC2CCCO2)COCCN1C(=O)Cn1ncnn1 O=S1(=O)CCCc2cccc(C(c3nnnn3C3CC3)NC34CC(C3)C4)c21 CCCC(C(O)C(=O)NCCCCO)NC(c1cc(C(N)=O)[nH]n1)=O C(C(C(=O)N1CCC(C(C)(C)C)C1)NC(=O)CCCC1CCC1)OCC.C(C)=O C=C(C)CC(C(=O)N1CCCC(CNC(C2CCC(F)(F)CC2)=O)C1)OC c1(OC)ccccc1C(C)=CC(=O)N(C1CCN(CC(=O)C(C)(C)C)C1)C N1(C(C(COC)C)=O)CCCC12CCC(NC(=O)Cc1nnc(S)n1C)CC2 C(=O)(CCCCCC#N)N(CCCNC(CC(=O)N(C)C)=O)C C(=O)(CCC(C)(C)C(=O)NC1CN(C(c2ccco2)=O)CC1OC)OC C1(CCNC(Cc2cccc(CC)c2)=O)CC(F)(F)CN1C(=O)CSCCOC CC(C)CC(=O)NCCC(=O)NC(C)CC1CN(C(=O)C(O)CN(C)C)C1 C(=O)(C1=CCOCC1)N1CCC(N(C(c2c(C)nc(C3CC3)s2)=O)C)C1 c1(CCN=C(NC(CC)C)NCC2CN(C)CCO2)nc2ccc(Cl)cc2[nH]1 c1(C(N(C(CNC(C2C(C(=O)OC)C2)=O)C)C)=O)ccccc1CN(C)C(C)C C1(NC(N(CC(c2ccc(Br)cc2)O)C)=O)CC2(CCC2)C1O C1(NC(c2cc(C)sn2)=O)CCCC2CN(C(c3nnn(C(C)C)c3C)=O)CC12 N1(C(C2C(C)C2C)=O)CCCCC(CNC(c2nn(C)cc2Cl)=O)C1 CCS(=O)(=O)c1ccc(CNC(C2CCC3C(CC2)C3(F)F)=O)s1 Cc1cc(NC(C2CC3CC3N2C(=O)CCC2CC2)=O)cc(Cl)c1 C1(OCC)CC(C(=O)NCC2(CF)CC2)C1.C1C(=O)N1.C1(C)CCC1.CCOC N1(C(C(=O)NC2C(C)CC(C)(C)CC2)=O)CCc2ncccc2C1 C1(C(C)(C)C)(CNC(Cc2ncc(C)o2)=O)CCN(C(=O)CCN(C)C2CC2)C1 C1(C(=O)NC2CCC(NC(c3cncc(C)c3)=O)C2)CN2CCC1(C)CC2 C12(C(N3CCC(F)(CNC(C(C)C(C)(F)F)=O)CC3)=O)CC3CC(C(=O)N1)C2C3 c1(C(C)=O)cc(C(=O)OCC(C2CCOC2C)=O)n[nH]1 C1(CNC(c2ccc(CC)[nH]2)=O)CC(NC(c2ccc(N)cn2)=O)C(O)C1 c1(N2CCC(C)C2CNC(c2ccc3nonc3c2)=O)ncnn2c(Br)ccc12 C=C(C)C(CC(=O)N1CC(NC(c2cc(Cl)ccc2CC)=O)CC(C)C1)OCC C(=O)(C1=CCOCC1)N(CCCCN(C)C(C1CN(S(C)(=O)=O)C1)=O)C C(=O)(C1c2ccccc2OCC1(C)C)NCCNC(C(CC=C)(C)C)=O N1(C(C2C=C(C)CS2)=O)CCC2(C=C(C(=O)N3CCOC(CC(C)C)C3)C2)C1 c1(C(=O)OC)cc(C(=O)NCC(C)(O)CNC(=O)Cc2cccnc2C)c(C)o1 c1(N2C3CC(CNC(C(C=CCCC)O)=O)C2CC3)cc(C)nc(S(C)(=O)=O)n1 CC(C)CCC(=O)NCC(=O)NC1CCC(N(C)C(C2C3CC3C3CC23)=O)CC1 c1(C(=O)NC2C(NC(C(CC#C)C)=O)C2)cnc(CC2CC2)nc1O C1(NC(=O)CN2CCC2)(CO)CCN(C(=O)C(c2ccccc2)F)C1 N1(C(C2(C)CCNC2=O)=O)CCC2CCC(C1)N2C(c1ccc2oncc2c1)=O O=C(CCCF)NC1CCC1CNC(=O)CC1(n2cccn2)CC1 C1(NC(=O)Cc2ccncc2Cl)CC2CCC1CC2NC(C1(O)CCCC1)=O C(CC1=CCN(C(=O)Cc2cnc[nH]2)CC1)NC(C(=Cc1ccccc1)OC)=O C(=O)(CC(C)C(C)C)N1C(C(C)NC(C(COC)COC)=O)CCC1 c1(C(N2C3CC(NC(C(CC)C)=O)C2CC3)=O)cccc2c1CCCN2 c1(C(N(CC(CC)NC(=O)CCP(C)(C)=O)C)=O)csc(S(C)(=O)=O)c1 N1(C(c2nn(CC)c(O)c2)=O)CC(NC(C23CC(CO2)C3)=O)CCC1C Cc1cc(C(N2CC=CC(NC(C3CC3F)=O)C2)=O)n(CC(F)F)n1 C(CC(CC)C(=O)NCC1CCCCN(C(=O)C(=O)NCC)C1)=CC N1(C(CN(C)CC)=O)CC2CCCC(C1)N(C(C1COCCN1C=O)=O)C2 C1(NCc2ccsc2)CS(=O)(=O)C1(C)C.C1(OC)CCOCC1N C(=O)(CC1OCc2ccccc21)NC(C)CC1=CCCCC1 c1(NC(c2cnc(NC(C3C(C4CC4)C3)=O)cn2)=O)cc(Cl)cc([N+](=O)[O-])c1O c1(C(N(C2CCN(C(=O)C(C)(C)F)CC2)CCOC)=O)cccc2cccnc12 C1(O)(CNC(CSC(C)C)=O)CCN(C(=O)CC2CCC2C2CC2)CC1 CN(S(=O)(=O)N1CCN(C2CCCCC2O)CC1)CC#N c1(C(=O)NCCN(CCOC)C(c2cnn(C3CCC3)c2)=O)ncsc1C C1(C(N(C(CNC(c2cc(C#C)cc(Cl)c2)=O)C)C)=O)CCN(S(N)(=O)=O)CC1 C1(C)(CC)CC(NC(=O)C=Cc2cc[nH]c2)CN1C(=O)Cc1cc(C)cs1 c1(CNC(CC(c2ccccc2)NC(C2(C)CCCN2)=O)=O)cccc(F)c1 c1(N(C(=O)NCC2CC(CC#N)C2)C)nc2ccc(Oc3ccccc3)cc2s1 C(C(C)CC(=O)NCC(CC(=O)N1CCCCCC1)C1CCC1)OC C(C)(C(=O)NC1CC(N)C1)NC(CSC(CC)C)=O N1(C(C(C)OCC(C)C)=O)CCCCC(N(C(=O)CCC2CCC2)C)C1 C1(NC(CCC=C)=O)CC12CCC(NC(c1nn(C)c(C(F)(F)F)c1Cl)=O)CC2 c1(C(=O)NCC2C(NC(C3N(C)C(=O)NC3)=O)C2)cnc(Cl)c(N)c1 c1(C(=O)NCCC(C)NC(=O)CC2CCCCCC2)cccc(Cl)c1 c1(OC)cn(CC(N2CC3CC(CNC(C4(O)CCC4)=O)C3C2)=O)c(C)cc1=O N1(c2n(CCCOC)c(C(c3cnccn3)C)nn2)C2CCC1CC(=O)C2 c1(C(=O)NC2(C(=O)NCCC(=O)N(C)C3CC3)CC2(C)C)cccc(O)n1 N1(C(C(C#N)C2CC2)=O)CCC2(CC1)CC2NC(c1ccc2cccnn12)=O c1(C(=O)NCCC(C)NC(C2C(=C)C2)=O)cnc2ccnn2c1N c1(C(C(N2CC(O)(CCNC(CCc3n(C)ccn3)=O)C2)=O)O)cccc(F)c1 c1(OC)ccc(C(N2CCCC2C(=O)NCC(C)N(C(=O)CO)C)=O)cc1 C(=O)(C(=O)N=S(C)(C)=O)NCC(CN(C(c1cc(COC)sc1)=O)C)C C12(C(=O)NCc3nc(CNC(CCC(=O)NCCC)=O)sc3)CCC(CC1)CC2 C=CCC(C)(C)CC(=O)NCC1CC(C)CN(C(c2cccc(C)c2C#N)=O)C1 c1(C(=O)NC2C(OC)CN(C(C34CCC(CC3)CO4)=O)C2)cc2cccnc2s1 c1(-c2ccc(C(C)O)cc2)ccc2ccc(C(N3CC4COCC4C3)=O)nc2c1 C12(NC(CC3CCC(=O)N3)=O)CCN(C(=O)C3=NOCC3)CC1C2 CC(CC(=O)N(C1CN(C(C2CCC2C#N)=O)CC1(C)C)C)C(F)F c1(CN(CCCn2cncn2)C)nc(-c2cccc(Cl)c2)nn1CCS(C)(=O)=O c1(C(N2CCCC(NC(c3n(CCC)ccc3)=O)CC2)=O)cc(Cl)c(F)cc1O C1(=O)C(C)CC(=O)NC2C(OC)CN1C2.C1(C(=O)OC)C2CCCCCC12 N1(C(C(CN(CC)CC)F)=O)CC(CNC(c2cn(CC)nn2)=O)C(C)(C)C1 N1(C(c2c(C(=O)OC)con2)=O)CCN(C(c2cc(C3CC3)ns2)=O)C(C)C1C CCC(CC(=O)N1CCN(C(=O)CCOC2CCC2)C(C)C1)CC(F)(F)F CC(C)CCC(F)C(=O)NCc1cn(CC(N2CCC(CO)C2(C)C)=O)nn1 C1(C(C(=O)NCC=C)N(C2CCN(S(C)(=O)=O)C2)C)CCC(C)(C)CC1 C1(C(=O)NC2CCCC(NC(c3nc(C)sc3)=O)C2)(N(C)C)CCCCCC1 N1(C(CCC(=O)OC)=O)CCc2c(C(=O)OC)n[nH]c2C1.C1(C)C(=O)OC(=O)N1 c1(C(N2CCCC(O)(CN(C(C(C)SC)=O)C)C2)=O)cnc2[nH]ncc2c1 C1(NC(Cc2c(C)nccc2)=O)CC2CC1N(C(=O)COc1ccc(Cl)nc1)C2 C#CC1(O)CC(C(N2CCC(O)(CN(C)C(c3c[nH]nc3C)=O)C2)=O)C1 C12(NC(CCC(C)(C)OC)=O)CCCC1CN(C(c1ccncc1Cl)=O)C2 N1(c2c(C)c(N3CCCc4c[nH]nc4C3)ncn2)CCSC2(CCOCC2)C1 c1(C(COC(C)C)C)cn(CCN(C)C(C2C(c3ccccc3)C2C)=O)nn1 c1(N(CCOC)CC)cc(Br)ccc1S(=O)(=O)NCC1CCC(OC(C)(C)C)C1 c1(CC)nc(Cl)c(C)c(=NCC2CN(C(=O)CCCc3nc(C)cs3)C2)[nH]1 N1(C(c2cnc(C)s2)=O)CCC2CC2(C(=O)N(C2CC2)C2CC2)CC1 C1(C(=O)NC(COCC)C(=O)NCC2C=CCCC2)COCC1(C)C CS(=O)(=O)c1ccc(N)cc1-c1c[nH]c2ccc(OCC(=O)O)cc12 C1(C(=O)NCC(CNC(C(C)(C)c2ccncc2)=O)(C)F)Cc2ccccc2O1 N1(C(c2nc(CCC)sc2)=O)CC2ON=C(CNC(c3csc(C)c3C)=O)C2C1 CC(O)C(O)CNC(c1[nH]ccc1CNC(C1(C#N)CC1)=O)=O C1(N(C(=O)COCc2cccc(CO)c2)CC)CCN(C(C2(F)CC2)=O)CC1 C1(C(C)NC(c2ccoc2Br)=O)CCN(C(=O)C=C2CCC2)CC1 CC1CC=C(C(=O)N2CCN(CCCNC(C3CCCNS3(=O)=O)=O)CC2)CC1 CCC(CC(C)C)C(=O)N1CCCCC1Cn1cc(O[Si](C)(C)C(C)(C)C)nn1 c1(C(=O)NCC2OCCN(C(C(c3ccc(C)o3)C)=O)C2)ccc(F)c(F)c1C c1(CC(=O)NC2C(NC(=O)Cc3ccncc3)CCC2)ccccc1C(F)(F)F C1(NC(c2cnn(CCC)c2C)=O)CCSC12CN(C(=O)CC(C)F)C2 N1(CCOC)CCN(C(=O)C(C)(C)C2CCCN2C(=O)CCC2CC2(C)C)CC1 C1(C(=O)NCCc2c(C)noc2C)CC12CCN(C(=O)CCC1CCC1)CC2 c1(C(=O)NCC(c2ccc(C)cc2)NC(CC(C)OC)=O)ccncc1F N1(CCCNC(=O)NC(c2cnns2)C)CCOCC1C C1(C)(C(N2CCC(N(C)CC)CC2)=O)CN(C(C2CCCC(=O)N2)=O)C(C)(C)C1 C1(CNC(Cc2c(C)cccn2)=O)CCCC2CN(C(c3cc(Cl)no3)=O)CC12 c1(C(N2CC(NC(C(C)NS(CC)(=O)=O)=O)C2)=O)cn(C)ccc1=O CCC(C)CC(C(=O)NCC12CCC(CC1)OC2)NC(=O)CC(C)(C)O N1(C(CN2CCC(OC)C2)=O)CCN(CC(C)C)CC1.c12nocc1C(=O)NC2 N1(C(C)=O)CCOC(C(=O)NCCCCN(C)C(C2CCNC2=O)=O)C1 C1(C2CCOCC2)(C(N2CC(COC)C(NC(C(C(CC)C)OC)=O)C2)=O)CC1 CCCCC(CN1CCOCC(C(=O)NCCCn2ccnc2C)C1)CC C1(C(N(C(CCNC(CC(=C)C)=O)C)C)=O)CN2CCN1C(C)C2 S(=O)(=O)(c1csc2ccccc12)N1C(C)CCC(NS(CCOCC)(=O)=O)C1 N1(C(C(c2ccnn2C)C)=O)CC2CCN(C(C3CCOCC3)=O)CC2C1 C(=O)(CCCCCCCC)N1C2(C(N(OC)C)=O)CC(C1)C2 C1(NC(C(C2CCC(O)CC2)(C)C)=O)CCCCC1CNC(c1scnc1Cl)=O c1(OC)cc(CN2CC3(CC3C(=O)Nc3cc(F)c(I)c(F)c3)C2)cc(I)c1O O=S(=O)(CCCCNS(=O)(=O)NC1CCCCC1)c1ncccc1Br C(=O)(C1=CCCCO1)N1CCC(CCC(C)(C)NC(C(C)CC2CCC2)=O)CC1 C(=O)(CC(C)C(C)(C)NC(=O)C(C)C1CCCC1)N(C(CC)COC)C c1(C(N2C(CNC(C(C(C)C)N(C)C)=O)CC2)=O)ccc2c(c1)CCO2 c1(CC(=O)NCC2CN(C(c3cncn(C)c3=O)=O)C2)cccc2ncccc12 C1(NC(=O)OC(C)(C)C)CC2CSCC(C1)C2C(=O)NCCC1CC1(C)C c1(CC)ccc(NC(CC2(CNC(C3(S(C)(=O)=O)CC3C)=O)CCC2)=O)nc1 C1(N(C(C=C(CC)C)=O)C)CCN(C(=O)CCN2CC(C)(OC)C2)C1 O=C1CC(C(N2CCCC(n3cc(CC4CCCCCC4)nn3)C2)=O)CCN1 Cc1cc(C)cc(C=CC(=O)N(C2CN(C(=O)C(C)SC(C)C)CC23CC3)C)c1 C=CCC(CC=C)C(=O)NC1CCC(NC(c2ncc([N+](=O)[O-])n2C)=O)CC1 C(=O)(CCCCCN(C)C)NC1(CC(N2C(COC)COCC2)=O)CCC1 CN1CCC(CC(=O)NC(C)(CNC(c2ccsc2Br)=O)CO)C1=O C(=O)(CS(=O)(=O)NC)NCC(CC)NC(C12CC(OC)C1C2)=O C1(CCCNC(c2cccs2)=O)CN(C(=O)CSc2ccccc2)CCO1 CN1CCOC(C(N2CC(CNC(c3ccccc3Cl)=O)C3CC23)=O)C1 N1(C(C(c2ccco2)NC(C2CCOC2)=O)=O)CCC2C(O)CC12 N1(C(C(CC)O)=O)CCCC(O)(CNC(c2ccc(CO)cn2)=O)C1 c1(C(C)C)ncncc1C(=O)NC1(CO)CCCCC1.C(C)(C)(C)NC(=O)O C(=O)(C(CCc1ccc(Cl)cc1)N1CCN(C(C2CCC2)=O)CC1)NCCSC O=C1CCC(CC(=O)NCC(C2CCOC2)NC(=O)CNS(N)(=O)=O)N1 C12(NC(c3nc(COC)oc3)=O)CC(C1)N(C(c1ccc(Cl)cn1)=O)C2 c1(C(C)C(=O)NCC2(O)CN(C(=O)CN3CC4CC4C3)C2)cncc(F)c1 c1(OC)cc(C#N)ccc1C(N1CCC(C)(CNC(c2ccc(Cl)cn2)=O)C1)=O Cc1cc(C(N2CCC(CNC(=O)COc3ccsn3)(CO)C2)=O)cn1C(C)C C=C1CCN(C(=O)C(C)CC=CCC)C(C(N2CCC2(C)C)=O)C1 CC(C)(C)C(CNC(=O)CC1CC1C1CC1)C(=O)NOCC1CCOCC1 N1(C(C(n2cnc(C#N)n2)C)=O)CCCC(C(N2CC(O)C(O)C2)=O)CC1 Cc1cc2c(C(=O)NCC3CC3CNC(=O)Cc3ncc(C)s3)ccc(C)c2[nH]1 C(=O)(C1=CCCCCC1)NC12CCN(C(c3sc(C)c(Br)n3)=O)CC1C2 C1(C(=O)NC2(C)CN(C(c3cc(CN4CCCCC4)on3)=O)C2)CCCOCC1 c1(C(=O)NC(C(C)NC(CC(CCC)O)=O)CO)c(C)ccc2c1CCCN2 N1(C(c2nc(COC)oc2)=O)CC2(C1)CN(C(c1ccc(O)nc1)=O)CC2CO CCC(C)(C)C(O)C(=O)N(C1CN(C(c2cnc(C(C)(C)C)nc2C)=O)C1)C C1(C(=O)NCC2(CNC(=O)CCF)CCCC2)CCCCC1N1CCCC1=O c1(CN2CC(C(=O)NCCc3ccccc3Cl)C(O)CC2)c(F)cc(Cl)cc1Br C(c1cn(C)cn1)=CC(=O)NC1C(C(=O)NC(CC)CCOC)COC1 c1(C(C)(C)C(=O)NC2CCCC=C2Br)ccc2c(c1)OCO2 CC#CCCCC(=O)N1CCC(NC(=O)Cc2cccc(NC(C)=O)c2)C1 c1(OCC(CN)O)ccc(C)cc1.c1(CCN2CCCC2)ccccc1.CO Cn1nc2c(c1O)CCN(c1cc(Br)c(C3CC3)cn1)C2 c1(OC)cccc2c1C(NC(c1c(C(=O)O)cc(Cl)cc1C)=O)CC(C)C2 c1(N2C(C)CC(C#N)C2)cc(=NC(=O)Nc2c(NS(C)(=O)=O)ccc(Cl)c2)[nH][nH]1 c1(NC(C2N(C(c3cc(C)c(F)nc3)=O)CC=C2)=O)cc(Br)c(F)cc1F Cc1cc(C(N2CCCC2C2CCN(C(C3(O)CC3)=O)C2)=O)cc(Br)c1 Cc1sc2ncc(C(N3CCC(CCNC(c4ccnnc4O)=O)C3)=O)n2c1C C(C(CN=c1[nH]c(N2CCCC(C#N)C2)nc2c1COC2)C(C)C)OC O=C(C1CCCc2c(O)cccc21)NCC1(O)CN(C(C2SCCCS2)=O)C1 N1(CCOC(C(C(=C)C)(C)O)=O)C(=O)NC2(CCCCC2C)C1=O C(=O)(C(C)(C)C(=O)NC(C1CCCN(C(c2ccc(Cl)cc2)=O)C1)C)NC N1(C(c2n(C)c(Cl)nc2)=O)CCC(C(=O)NC2CC3OCCCC23)C12CC2 c1(NCC2(SCC)CC2)[nH]c(=NCCCc2ccco2)nc2sccc12 C(=O)(CCC(=O)N1CCC(COC)(NC(C2CCCC2F)=O)C1)NCCC C1(F)(C(=O)NC(C)(C)C)CCN(C(=O)Cc2sc(O)nc2O)CC1 CCS(=O)CC(=O)N(C1CN(C(=O)Cc2csc(Nc3ccc(Cl)cc3)n2)C1)C c1(C(=O)NC23CCN(C(=O)CN4CCOCC4=O)CC2C3)ccc2c(n1)CCC2 CC(C)(C)C(C(=O)NCCCNC(=O)CC(F)(F)Cl)N1CCOC1=O CN1CCN(C(C2CCN(C(=O)C3CCSCC3)O2)=O)CC1CO C1(C(=O)NC2CCCCC2F)CC12CCN(C(c1cccnc1O)=O)C2 c1(C(=O)NCC(CC(=O)NC(C)CCC2CC2)C)coc2ccccc12 c1(OC)ccc(CC(C)C(=O)N2CCCC2CCCNC(C2(CO)CC2)=O)cc1 C1(NC(c2cc(C(C)C)on2)=O)CCN(C(C2CC(C)(O)C2)=O)C1C1CC1 Cc1cn2c(C(=O)Nc3ccc4occc4c3)cnc2s1 C(=O)(C(F)(F)CCc1ccccc1)NCC(CNC(C1CC(C#C)(O)C1)=O)OC CCC(C(=O)OC)C(=O)NC(C(=O)NCC1CC1[N+](=O)[O-])C(C)(C)C C1(CNC(c2coc(Cl)c2)=O)(NC(=O)C(=C2CCCCC2)F)CCCC1 c1(-c2scc(OC)c2)ccccc1C(=O)NCC1CCC(=O)N1C C1(CNC(C2(C(=O)OCC)CCC2)=O)CN(C(c2coc(C3CC3)n2)=O)CC1C C=CC(CCC)CC(=O)N1CC(CC(F)C(=O)NC(COC)C(C)C)C1 C(CC(=O)NCCC1C2CN(C(C3CCC(=O)N(C)C3)=O)CC12)(C(C)C)OCC C(CCC(C)NC(=O)C(C)NC1CCOCC1)NC(C1(CCCC)CCC1)=O c1(NC2CCN(OC)CC2)ccc(S(=O)(=O)N(CC(C(C)C)N(C)C)C)c(Cl)c1 c1(C(=O)OCC)cc(S(C)(=O)=O)cnc1NC(=O)N(CC)CC1CC(F)(F)C1 c1(C(=O)NC(C2CCCCO2)C)c(NC(=O)COC(F)(F)F)cccc1F c1(C(=O)NC2CC3(C2)CN(C(=O)COCCF)C3)cc([N+](=O)[O-])cc(Cl)c1Cl c1(C(=O)NC23C(CN(C(C4(SC)CC4)=O)C2)CCC3)ccn2c(O)nnc2c1 C(=O)(C(C)(C)CS(N)(=O)=O)NCC1C(C)CCN1C(c1cc(F)n(C)n1)=O Cc1cc(F)ccc1C(=O)NCC1CCCN1C(C1(C#N)CCCOC1)=O C(=O)(CC(C(F)F)N1CCOCC1)NCC1CN(C(c2c(C)noc2C(F)F)=O)C1 N1(C(c2cn(CCC)nn2)=O)CCC2(CC2)CC1C(N1CCN2CCC1CC2)=O c1(C(=O)NC(C2CCCCC2)CNC(c2c(CC)nc[nH]2)=O)cc2n(n1)CCC2 c1(NC)cnccc1C(=O)N(CC(C)C(N1CCCCC1C(F)F)=O)C CCCC(F)C(=O)NN1CCC(C)CC1.c12cnncc1NC2(C)C.OC C=CC(C)(CCOC)C(=O)NCC1CC2(CCC2)CN1c1nccc(C)n1 N1(C(C2(CC)CCCCO2)=O)CC(CN(C(=O)CC(C)O)C)C2(CC2)C1 CN1CCOC(C(=O)NCCCNC(c2cnc(-n3cccn3)cn2)=O)C1 C(=O)(CC1=CCN(C)CC1)N1CCC(CN(c2ccc(Cl)cc2C#N)C)CC1 C#CCCCCC(=O)NC1COCC1N1CCN(C(C2CN(C)C2)=O)CC1 c1(SC)nc(NC2CCN(C(C3(F)CCOC3)=O)CC2F)cc(OC)n1 CCC(CC)C(C(=O)N1CCC(O)C(NC(c2cnsc2)=O)C1)OC C1(OC)(CNC(=O)Cc2c(C)n[nH]c2C)CCN(C(C2CCN(C)CC2)=O)C1 N1(C(CCC2C(C)C2)=O)C2CCC1C(CNC(c1ccccc1SCC#N)=O)C2 N1(C(CS(CC)=O)=O)CCC(CO)C(NC(=O)C2CC2)C1 C1(C(N2CCN(CCC)CC2)=O)CC2CC1CC2NC(C1CCN(CC)C1)=O C=CC1CC(NC(C2(CCC=C)CN(C(=O)CC3CNC(=O)O3)C2)=O)C1 C1(C(N(C2CC2)CC2N(C(CNC(C)=O)=O)CCC2)=O)CC(=O)N(C)C1 N1(C(C(CC)CC(C)C)=O)CCCC2(CCCCC2NC(C)=O)C1 c1(C(=O)NCC(CO)NC(C(CSC)C)=O)ccc2c(c1F)CCC2 C1(C(N2CCC(C(C)(C)NC(c3cnccc3Cl)=O)C2)=O)Cc2nncn2C1 c1(C(N(C2C(C)COCC2)C)=O)[nH]nc2ccncc12 c1(N2C3CC(CNC(c4c(C)cn(C)n4)=O)(OC3)C2)ncnc2c1c(Br)nn2C c1(C(N2CCC(C)C(NC(c3ccc(C)o3)=O)C2C)=O)ccc2c(c1)CCCS2 c1(C(N2CCC(C(CNC(C(NOC)=O)=O)C)CC2)=O)ccc(OC)cc1C N1(C(CCN(C(CC2COCC(C)O2)=O)C)=O)CCCCN(C)CC1 S(=O)(=O)(CCC(C)(F)F)NCc1c(-c2c(C(C)C)cccc2)cccn1 C1(C(=O)NC2CC(NC(c3cc4scc(C)c4[nH]3)=O)C2)C2Cc3ccccc3C12 C(=O)(CC(C)(C)C(=O)NCC1CC(O)(CNC(C2CC3C=CC2O3)=O)C1)OC Cc1cnc(C(=O)NCc2occc2C(=O)NC2C3CCCC23)c(F)c1 C1(F)(CNC(C2C=CCCC2)=O)CCN(C(C2CC(O)C2)=O)C1 C(N=c1cc(C)[nH]c(=NCC=CCCOC(C)C)[nH]1)C1N(S(CC)(=O)=O)CCC1 C1(CC=C)(NC(C2CC2c2cnc[nH]2)=O)CCCN(C(=O)CS(N)(=O)=O)C1 C1(CNC(CCC(C)C)=O)CCN(C(C23C(=O)C4CC2C3C4)=O)CCC1(F)F N1(C(C(CCC)NC(=O)C=CCN2CCCC2)=O)CCS(=O)C(C)C1 Cn1nccc1C=CC(N1CC2CC1C2C(=O)Nc1cncc(Cl)c1)=O CC(CCN=c1ncc(Cl)c[nH]1)NC(c1ccnc(C2CC2)c1)=O N1(C(c2ncc3ccccc3n2)C(=O)NC)CCCCCC1C1CCCO1 c1(C(N(CCC(=O)NCC(O)(C2CC2)C2CC2)CC=C)=O)cc(C)no1 c1(-n2c(N3CCCC(O)C3)nnn2)cc(Cl)c(Br)cc1Cl C1(OCC(=O)NC(c2cccnc2)C(=O)NCC2C(C(N)=O)CC2)CCOCC1 Cc1ncc(C(=O)NC2CCC2C(N2CCN(CCOCF)CC2)=O)cn1 C(CNC(C1(C#N)CCCO1)=O)(C(C)(C)C)NC(c1nc(C(C)C)sc1)=O Cc1ccc(-c2nc(-c3cncs3)nn2-c2c(C)noc2C)c(F)c1F C1(F)(CNC(=O)C=Cc2cc[nH]n2)CCN(C(c2cc(Cl)no2)=O)C1 C1(C(N(CCCC(C)O)C)=O)CC2CN(C(c3cnn(C)c3C#N)=O)CC2C1 c1(C(N2CCC(N(C(c3onc(CCOC)n3)C)C)C2)=O)cnc2[nH]cnc2c1 CC(C)(C)S(=O)(=O)c1ccc(NC(=O)Cn2nnc(C3CC3)n2)cn1 CCCC(C(=O)N(CCCCNC(=O)C(N)=O)C)OCc1ccccc1 C1(C(=O)NCCN(C)C(c2cccc(O)n2)=O)CC(c2cnn(C)c2)=NO1 CC1CN(C(=O)CC2CCCC2)CCC1CNC(C1(C)CC(F)C1)=O c1(C(N(C)CC2N(C(C(C)NC(C)=O)=O)CCC2)=O)c(C)noc1N N1(C(C(C)SCC)=O)CCC(c2cc(CNC(C3CCC(C)C3)=O)on2)CC1 c1(C(=O)NC)cccc(C(=O)NCC(F)CNC(=O)CSc2ccccc2)n1 C1(C(=O)NCC2CN(C(C3(C4CCCO4)CCC3)=O)C2)CC2CCCN2C(=O)N1 N1(C(CCCC=C)=O)CCC2(CC2NC(C23CCC(C2)C3(C)C)=O)C1 C1(CCNC(c2ccc(Cl)cn2)=O)CCc2ccccc2C1 N1(C(C(c2c(C)cccc2)(F)F)=O)C2CCC1CC(N1CCCCC1)C2 Cc1cnc(CCNC(=O)C(C)(C)C2CCCN2C(=O)C(O)C2CC2)nc1 C(=O)(C(CCC(C)C)NC(C)=O)NC1CC(NC(CC2(OCC)CCC2)=O)C1 C=C(C)CC(C)C(=O)NCC1CCN(C(c2cnc(C)n2-c2ccccc2)=O)CC1 C1(CNC(C2CC(=C)C2)=O)CCCCN1C(C1CC(OC)(OC)C1)=O C(N=c1ccnc(NC2CCCC(F)(F)C2)[nH]1)c1cncc(C)c1 Cc1ccc(CCC(=O)N(CCCCC(=O)OC(=O)OC(C)(C)C)C)cc1 C(=O)(CCC(O)C(C)(C)C)NCC(C)N(C(c1c(OC)nn(C)c1)=O)C C1(c2ccc(OC)cc2)CCN(C(=O)CN2CCC2)CC1NC(=O)CN(C)C N1(C(C2(N)CCCCCC2)=O)CCOC2(CC1)CCS(=O)(=O)C2 C1(CNC(c2scc(C)c2)=O)CCC(C)(C)CN1C(C1CCCN1C1CC1)=O c1(C(=O)NC(CC)CC(=O)N2CC(C(C)OC)C2)ccc(O)c(F)c1 Cn1ncc(C#N)c1C(=O)NC1C=CC(CC(=O)NC(CO)CCO)C1 C1(c2nnnn2C2(C)CC2)(NCC2C=CC(C)(C)CC2)CC2(C1)CC(C)(C)C2 Cn1cc(CC(=O)NCCCOCCNC(=O)CN2CSCC2=O)c(C(F)F)n1 C1(CC)CCN(C(c2c(C)cnn2C)=O)C1CNC(=O)CNC(=O)NC c1(OCC)ccc(C(=O)N(CCC(C(C)C)NC(=O)C(CO)N(C)C)C)cc1Cl N1(C(C=CCC)=O)CCN(C(c2ccc(C(C)C)c(F)c2)=O)CCC1C C1(NC(C(Br)=C(C)C)=O)CC2CC(NC(C3C4C5CCC(C5)C34)=O)CC12 C1(N(C(C2(C(=O)OC)CC2)=O)C)CNCC1F C(=O)(C(O)CC(N)=O)NCC1C(CC(=O)NCCCCC2C(C)C2)C1 N1(CC)CC(C(=O)NC2CCC2NC(=O)Cc2cccc(F)c2)CCC1=O C1(CCC(=O)OC2CSC2)CCCN(C=O)C1.C(=O)(CCCc1ccccn1)CC c1(C(C)(C)C#N)cccc(C=CC2CCCC2)c1 c1(OCC(=O)Cc2ccccc2F)ccc(Cl)cc1Cl C(C(COC)CC(=O)N1CC(CNC(c2ccccc2O)=O)C(O)C1)OC c1(CN(C(=O)NC23CC(C(=O)OC)(OC2)C3)CC)cnc(C)c(C#N)c1 c1(C(=O)NCC#CCNC(C(C2CC2)SC)=O)ccc(C)c(-c2cccs2)c1 N1(C(CN(C)S(N)(=O)=O)=O)CCC2(CCN(C(=O)CC3CCOC3)C2)C1 C(CC(C(=O)N1CCCC(CN(C)C)C1)NC(C1CN(C2CC2)C1)=O)=CC C(C(COC)CC(=O)NC1CC(NC(=O)C(C(C)(C)C)OC)C1)OC N1(C(C2C(COC)CC2)=O)CCC2(NC(=O)CSc3n[nH]c(O)n3)CC2C1 C#CCCCCCC(=O)N1CCC(C(=O)NCc2noc(COC)n2)C1(C)C N1(C(C(C2CC2)OCC)=O)CCCC(N(C(C2CC(=O)N(CC)C2)=O)CC)C1 C(=O)(CCC(C)(C)C)N(C)CC1CCCN(C(=O)CC2COCCO2)C1 CC1=NOC(C)(C(=O)N(CCC(=O)NCCN2CCCCC2C)C)C1 C(N=c1nc2sccc2c(NCC23CCCCC2C3)[nH]1)C1(C(N(C)C)=O)CCC1 c1(OC)cnccc1C(=O)N(C(C)CNC(=O)C(C)(O)Cc1ccccc1)C CCC(C)(CNC(=O)C(COC)N(C)C)C(=O)NC1(CCCCO)CC1 C1(C(=O)NC2CC(C)(C)OC2)CCOCCN1C(c1ncccc1N)=O c1(OC)ccccc1C(=O)N(CC(O)CNC(=O)Cc1ccsn1)C Cc1ncccc1CCC(N1CC(c2cnn(C)c2)C(N)C1)=O CC(Cn1ccnc1)C(=O)NC1CC1NC(=O)CSCC(F)(F)F C(=O)(C(C)CC(C)C(C)=O)NC1(C(=O)NC2(CCC)CCC2)CC(CO)C1 C(C(N=[N+]=[N-])C(=O)NC1C(C(N2CCC(CC)(CO)CC2)=O)C1(C)C)OCC C(=O)(C(CC(F)F)NC(=O)CP(C)(C)=O)N1CC(CC)OCC1 Cc1nc2c([nH]1)CC(NC(=O)C(F)(F)c1ccn(C)n1)CC2 C1(NC(C2(CNC(c3c(CC)nccn3)=O)CC2)=O)CN(C)CC1(C)C c1(C(CC(=O)N(C)CC2CN(C(COCC)=O)C2)C)cccc(OC)c1 C(C(C)C(F)C(=O)NCCc1ccon1)NC(c1c(CC)nns1)=O c1(N(CC(CC)C)C)nc(N(C)CC2CCCO2)nc2ccccc12 N1(C(c2c(C)cc(CO)o2)=O)C2CCCC1CN(C(=O)CC1(C#N)CCC1)C2 C12(NC(c3c(Cl)cnc(C)n3)=O)CCCN(C(=O)C#CC(C)C)CC1C2 c1(OC)cncc(C(=O)NCC2CCCN(C(c3cc(O)cn3C)=O)CC2)c1C Cc1cnc2c(cnn2CC(=O)NC(C)CNC(c2cc(CC(C)C)on2)=O)c1 C(C)(CC(=O)N(C1CN(C(c2c[nH]nc2Br)=O)C1)C)OC CCCCC(C)C(=O)NC1CN(C(=O)CN(C)S(=O)(=O)N(C)C)CC1F C(CCCC(CO)NC(c1c[nH]nc1C(F)(F)F)=O)NC(=O)Cn1cnnc1O C1(C)(c2ccc(CNCc3c(O)ccc(C)c3)cc2)CC(C)(C)OC1=O C=C(C)CC(C(=O)NC1(CO)CCC1)NC(=O)C(C)=C(C)CC C12(NC(=O)Cn3ncnn3)CCCC(CN(C(c3ccc(C(F)(F)F)[nH]3)=O)C1)C2 c1(C(N2CC=CC(NC(C3CCn4nncc4C3)=O)C2)=O)ccc2cncn2c1 C1(C)(C(N(CCCCC(=O)NC)C)=O)CCN(C(=O)Cc2ccoc2C)CC1 CC(C)C(O)CC(=O)N1CCC(N(C)C(c2ccsc2Br)=O)C1 n1(CC)ccc(C(=O)NCC(=C2CN(C(C3CCC3(C)C)=O)C2)F)n1 c1(C(=O)NCC2OCCN(C(CC(CC)C)=O)C2)cc(NC)cnc1C C1(C(=O)OC)CC(NC(=O)CC(c2ccccc2)OC(C)=O)CS1 N1(C(C2CCN(C(COCCOC)=O)C2)=O)CCCC(O)(CO)C1 c1(NC(c2cc(C)c(C)cc2Br)c2n(CCC)nnn2)cc(Br)c(C)cc1OC C1(C)(C(=O)OC)CN(C(=O)C(=O)NCCC2CC(SC)C2)CC1(F)F C1(CNC(c2cc3n(n2)CCO3)=O)CC2(CCC2)CN1C(=O)CCOC1COC1 CC(F)(F)C(Cl)CNCCN(c1ccccc1)C(C=Cc1ccc(C(=O)O)o1)=O C(C(CC(=O)NCC(C)(C)CC1CC1)NC(=O)CCOCCN(C)C)OC C1(OC)CC(NC(c2cc(C)nc(O)n2)=O)CN(C(C2(C)CC(C)C2)=O)C1 CC(C)(O)C(F)C(=O)N1CCCC1C1CCN(C(C2CCCC3(CC3)C2)=O)C1 C1(NC(C(C)OC)=O)CCCC(CNC(=O)C(c2cccc(C)c2)F)C1 CC1(C)CCC(CNC(C2(CNCC3(O)COC3)CC2)=O)CC1 Cc1nc2ncccc2cc1CCC(=O)NC1CN(C(=O)Cc2csnc2C)C1 c1(CN(C(CF)CF)C)cc(Br)c(O)cc1F CC1(C)CN(C(C2CCCC2C(F)F)=O)CC(CNC(=O)COC2CCCC2)O1 c1(C(=O)NCC(N2CCCCC2=O)C)cnc2[nH]c(O)nc2c1 N1(C(CC2CCN(C)C2=O)=O)CC2(CCC2)CCC1CNC(=O)C1=CCC1 CC(C)CCC(C(=O)NC1CN(C)C(C)(C)C1)NC(C1CC(=O)C12CCC2)=O n1(CC(=O)N(CC(CNC(C(CC)OC)=O)O)C)nc(C(F)(F)F)c(Cl)c1C c1(OC)ccc(CCC(=O)N(CCNC(C2CC(C)OC2C)=O)CC2CC2)cc1 C(=O)(CCC(F)(F)Cn1cc(CNC2CCOC2)nn1)NC(CC=C)C1CC1 C(=O)(C(F)(F)Sc1cnn(C)c1)NCCN(C(=O)CCc1ccc(C)s1)CC c1(NC(CC)=O)cccc(C(c2cccc(OC)c2)N2CC3C(N)C3C2)c1 C1(O)(CN(C(C(C)(C)SC)=O)C)CCN(C(=O)CCSCc2ccccn2)C1 C(c1ccccc1C)=CC(=O)NC1(C(N2CC(C(=O)NCC)C2)=O)CCN(C)C1 C1(C(=O)NC2(CCCNC(C3(C)CC(C)(C)C3)=O)CC2)CC2CCC(C1)C2=O c1(C(=O)NC2(C(N3CCCC(COCC)C3)=O)CCCC2)cc(F)cc(N)c1F n1(C(C)C)cc(Br)c(C(=O)NCC2CN(C(=O)CC3(C)CC3)CCO2)n1 Cc1nc(C)n(CC(N2CC(NC(=O)Cn3ccccc3=O)C(C)C2)=O)n1 c1(C(N2CCC(O)C(C(N3CCCC(Br)C3)=O)C2)=O)ccc(F)nc1F C1(N(C(=O)Cc2ccccc2C(F)(F)F)C)CC2(C1)CC21CCC1 N1(c2nc(N3CC4C(N(C)C)C4C3)c3c(n2)scn3)CC23CCCC2(COC3)C1 Cc1ccc(Cl)c(C(N2CCCC(CN(C(=O)CNC(N)=O)C)C2)=O)c1N C#CCCCCCCNC(C1CCCCN1C(c1ccns1)=O)=O CN=c1nc(N2CCc3cc(C)cc(C)c3C2)[nH]c(=NCCN(C)C(C)=O)[nH]1 Cc1cn2c(n1)CN(C(=O)CC1(N(C3CC=CC3)C)CC1)CC2 Cc1ccc(C(=O)NCC(C(=O)NCCCSC(F)F)N(C)C)s1 N1(C(c2c(C)nn(CC(F)(F)F)c2)=O)CCOCC(NC(C2CCN(C)C2)=O)C1 C(=O)(CC(CC)CCCC)N1C(C)(C(N2CCN(C(=O)OCC=C)CC2)=O)CC1 c1(C(N(CCCNC(C2(C)CC2(F)F)=O)C)=O)c(N)cc(Cl)nc1Cl N1(C(C2N(C(C(COCC)(C)C)=O)C(C)C2)=O)CC2C(C1)C2(C)C Cc1cc(C)c(C(=O)NCC(C(=O)NCCC(C)N2CCCC2)N(C)C)s1 CC(CC(=O)NCC1CN(C(C2(C)CCCC2)=O)CC1C(F)(F)F)P(C)(C)=O c1(C(=O)OC)cccnc1C(N1CC2CC1C2NC(C12CC(CC(F)F)(C1)C2)=O)=O c1(OC(C(=O)NCC(C)(CO)NC(=O)CC=C(Cl)Cl)(F)F)ccc(Cl)c(F)c1 C1(NC(C(C(CC)C)OC)=O)CCCN(C(c2cncc(SC)c2)=O)CCC1 c1(-c2c(C)cc(O)cc2)cc2cc[nH]c2cc1C(=O)NC1CNC(=O)C1(C)C C#CCCCCCCC(=O)N1CCC(NC(=O)CSCc2ccccn2)C1 C12(C(N3C(CNC(C4(NC(N)=O)CC4)=O)CC(OC)C3)=O)CC1COC2(C)C c1(C(N(C2CC(NC(c3c(CCC)nco3)=O)C2)C)=O)ccc2c[nH]nc2n1 N1(C(c2cc(C(C)C)on2)=O)CCC(NC(=O)CN2CCCC2=O)C(C)(C)C1 N1(C(C(CC)CC(C)C)=O)CC=C(C(C)(C)C(=O)NC(C)C(O)C(F)F)C1 c1(C(C(=O)NCCCCCC)N(C2CCCC(O)C2)C)cn(CC2CC2)nc1C N#CC1CC(F)(F)CN1Cc1c(-c2ccc(C(=O)N)s2)cccc1.N1CCCC1 C(C(C)C(=O)N(CC(C)(C)CNC(C1CCC(C)O1)=O)CC)OCC N1(C(C(CC)NC(C)=O)=O)CC2CCC(C(=O)NC(CCF)C(=O)OC)(C2)C1 Cc1cccc(C(N2CCN(C(c3csc(Cl)c3)=O)CC2CO)=O)c1Cl C(CNC(c1cnn(CCC(F)(F)F)c1)=O)(C(C)C)NC(CN(C(=O)OC)C)=O c1(C(=O)NC(C2(O)CN(C(=O)COCCF)C2)C)cnc(C2CCOC2)s1 Cc1cc(C(=O)NC(C)CCCCNC(c2n[nH]c(C)c2O)=O)sc1C C(=O)(CCCCCN(C(=O)C1=C(Cl)CCC1)C)NCC1(CCOC)CCC1 Cc1cccc(C)c1C(C(N1CCC(O)C(C(=O)N=c2nc[nH]s2)C1)=O)C1CC1 c1(C(=O)NCC(C)CCO)cc2nc[nH]c2cc1[N+](=O)[O-] C1(C(=O)NCC2(C(=O)NCC3CCCSC3)CC2)C2CC3C(C2=O)C13 N1(C(C(C)(C)SC)=O)CCC2(CCCC2NC(=O)C(CO)c2ccccc2)CC1 C1(CNC(c2c(SCCC(=O)OC)cccc2)=O)CC2CCCCC2O1 c1(CCC)noc2nc(C3CC3)cc(C(=O)NC3CCCC3O)c12 C1(NC(c2c(C)cco2)=O)CN(C(=O)C(C)n2ccnc2)CC2(CC2)C1 C=CC(C)C(C)C(=O)NCCC(N)COC c1(CC(C)N(C)C)ccc(Cl)cc1.C12(CC(NC(=O)OC(C)(C)C)C1)C(=O)N2 CC1CC2CN(C(=O)Cn3nc(C(F)F)cc3C3CC3)CC2N1C(=O)C(O)CF C(=O)(C(F)C(F)(F)F)NC1C(NC(=O)CNC(c2ccncc2)=O)CCCC1 c1(C(=O)NC2CCCC(NC(C3CCOC3)=O)C2)c(-n2ccnc2)cccc1Cl CC(=O)CCN=C(NCCN1CCOCC1C)NCC1CC1(Cl)Cl N1(C(C2CCN(C)CC2)=O)CCC2(CC1)CCN(C(C1CCCOCC1)=O)C2 Cc1cc(=NCc2ccncc2N)[nH]cc1S(=O)(=O)NCC(CC1CC1)CO C=CCCCCCC(=O)N1CC2CC1(CNC(c1n[nH]c3c1CCC3)=O)C2 Cc1cc(Cl)nc(N)c1C(N1CC(NC(=O)C(C)(C)n2cnnn2)C(C)C1)=O C1(NC(c2c(CC)onc2)=O)CN(C(=O)CCOCCOC(C)=O)CC1C1CC1 Cc1cn(C)nc1C(=O)NCC1CCN1C(=O)C(C)(C)c1cnsc1 CCCC(CC1CCCC1)C(=O)N(CC(C)N(C(=O)Cc1cccc(Cl)c1)C)C CC(C)CC(C(=O)NC1CCCSCC1)NC(c1ccns1)=O C(=O)(C1CCCCc2ccccc21)N1CCC(O)(CNC(C(C=C)(C)C)=O)C1 C#Cc1cccc(C(=O)NC(C)CNC(c2nc(CC)oc2C)=O)c1Cl C12(NC(=O)COc3ccsc3)CCC(NC(C3(O)CCOCC3)=O)(CC1)C2 c1(CNC(C2CCCC3CNCC23)=O)cccc2c1OCCCO2 N1(C(C2(CC=C)CCC2)=O)CCCC2(CC(NC(c3cc(C)sn3)=O)C2)C1 C(=O)(C1CCc2ccccc21)NCCN(C(=O)C=CCOC(C)(C)C)C(C)C C1(NC(c2c(CC(C)C)n(C)nc2)=O)CC2CC1N(C(c1csnc1C)=O)C2 N1(N(c2c(C(C)=O)cc(C)s2)C)CC2CC1CN2C.c1(C=O)ccc(I)c(O)c1 Cc1ccncc1C(N1CCC1CNC(=O)C(C)(O)Cn1ccccc1=O)=O N1(C(c2cc(C(C)(C)C)[nH]n2)=O)CCN(C(=O)Cc2ccco2)CC1C1CCC1 C=C(C)CN=C(NCc1ccc(C(F)(F)F)s1)NCC(C)(O)CC C1(CNC(c2nc(Cl)c(Cl)s2)=O)CN(C(=O)Cc2c[nH]nc2O)CC1O c1(CN2CC(OC)C(NC(c3ncccc3F)=O)CC2)ccc(F)c(F)c1F C(=O)(CCCC(=O)N(CCCN(C)C)CCNC(c1ccc(F)s1)=O)OCC c1(C(=O)NCCCC(C)NC(=O)C(N2CCNC2=O)C)ccc(NC=O)cc1 C(=O)(C1=COCCO1)NCC(C1CCOC1)NC(CCc1cc(C)on1)=O c1(C(C)=O)ccc(S(=O)(=O)N2CC(F)(C(=O)Nc3cccnc3C#N)C2)cc1 C1(C)(C(N2C(c3c(C)cccc3)CCC2)=O)CCCN(c2ncc(Br)cn2)C1 c1(NC(CC(CNC(C2(COCC)CC2)=O)O)=O)ccc(F)c(C)c1 C12(CNC(c3ccc(C(F)(F)F)o3)=O)CCC(CC1)N2C(=O)C(F)(F)C1(O)CCC1 Cc1ccc(C)c(NC(=O)CN(C)CCN(C)C(n2nnc(C3CC3)n2)=O)c1 C(=O)(N=c1cc2n([nH]1)CCCN(Cc1ccccc1)C2)NC(CC)(C(N)=O)C(C)C C1(CNC(C2C(C)(C)C2)=O)CN(C(c2occc2F)=O)CCC12CCOCC2 CC1(C)CCC(F)(F)CC1C(N1CC2CCCC(C1)N2C(C1CCSC1)=O)=O c1(CCC(=O)N(C)Cc2cn(CC(COC)O)nn2)cc(OC)ccc1[N+](=O)[O-] N1(C(c2ccc(CC(=O)OC)cc2)=O)CCN(C(C2(C)CC2F)=O)C2(CCC2)C1 N1(C(C(c2n(C)ncc2)O)=O)C2CCC(C2)C1CC(=O)NCC(=O)NCCO c1(C(n2cc(CCCCNC(C3(F)CC=CCC3)=O)nn2)C)cccc(Cl)c1 N1(C(C2C(C)CCOC2)=O)CC(C)(C(=O)NC2CC(CC(C)(C)C)C2)CC1(C)C C1(CNC(C2(C)COC2)=O)CC2(CCN(C(=O)C=Cc3cccs3)CC2)CO1 C1(NC(CC2(CSC)CC2)=O)CN(C(C2(CC(F)(F)F)CC2)=O)CC1C C1(CC(=O)NCC2CC(CNC(COCC(N3CCCC3)C)=O)C2)COCCO1 c1(NCc2cnn(CCC)c2C)ncc(C2=COCC2)cn1 c1(C(C)C)nc2[nH]ccc2c(=NCCC2CCN(C(C3CC34CC(O)C4)=O)C2)[nH]1 Brc1ccc2nc(CCCNc3cccc(OC4CCCC4)c3)[nH]c2c1 N1(C(CCC(=C)Cl)=O)CCCCC2(C1)CN(C(C1CC3CCC1O3)=O)C2 CCCC(CC(C)C)C(=O)N1CCC(C(=O)N(C(C)CC(C)C)C)C(C)C1 Cc1cccnc1C(=O)NC1CN(C(=O)CC2(C)CC2(Cl)Cl)CC1C(F)F C(=O)(C1=NOC2(CCC2)C1)N1CCN(CC(C)NC(C=C(C)C)=O)CC1 Cc1nc(NCc2ncn(C)n2)cc(N(C(C)C(c2ccccc2F)O)C)n1 c1(N(CC(CNC(C(CCC)n2cncn2)=O)C)C)cccc(F)c1C#N c1(C2(C(=O)NCCCNC(C3CCSC3)=O)CCCC2)cccc(F)c1F CC(C)(CC(=O)NCC1CC(O)C(O)C1)NC(=O)Cc1ccc(F)nc1 N1(C(Cc2cccc(SC)c2)=O)CC(CNC(C2C=CCC2)=O)C(F)(F)C1 c1(CC(=O)NCCC(C(C)C)NC(CCCCOC)=O)ccc2ccccc2c1 Cc1cnn(C)c1CC(=O)NCCc1n[nH]cc1C(N1CC(CF)C1)=O c1(C(=O)NC2CCCCC2CN(C(c2csnn2)C)C)ccc2[nH]ccc2n1 N1(C(CCC(N)=O)=O)CCC(F)(CNC(C2CC2c2ccsc2)=O)CC1 C1(CNC(c2c[nH]c(=NC)o2)=O)N(C(=O)CC2CC2C)CCCC1(C)C c1(C(N2C(CC(=O)NCc3ncc[nH]3)COCC2)=O)ccc([N+](=O)[O-])cc1F C1(C(=O)NC(CNC(CCCC2C(C)C2)=O)(C)CO)CC2(CCC2=O)C1 N1(C(CC(C)OC)=O)CC(NC(=O)Cc2cncn2C)C(N=[N+]=[N-])C1 N1(C(c2c(CC)cco2)=O)CC2CC1CN(C(=O)CC1OCCC1(C)C)C2 C12(CNC(C3(CNC(C4N(CC)CC4)=O)CC3)=O)CCCC(CO1)C2 C(CC1CCC1)(C(=O)NC1C=CC(CC(=O)NCC2(C)CC2C)C1)OC C1(CNC(CC(C)C2CC2)=O)CC2(CO1)CN(C(=O)Cn1ncnn1)C2 C1(C#N)(C(=O)NC2C=CCC(C(=O)NCCCc3n(C)cnn3)C2)CCCCC1 C1(C(=O)NCC(C(C)(C)O)O)CCC(C)(C)N(C(C2CC3CC2CC3=O)=O)C1 N(C(=NCC1CC1)N1CCC2(CCOCC2)CC1)CN1C(=O)CCNC1=O C1(O)(CN(C(CC2ON=C(C)C2)=O)C)CCN(C(C2(C)CC2)=O)C1 N1(C(CCc2c(C)ncs2)=O)CCCC(F)(CNC(c2coc(Cl)n2)=O)C1 c1(C(=O)NC2C3CC(NC(=O)Cc4ccccc4F)CC32)coc2ccccc12 C(=O)(C1=CCCCCC1)NCCCN(C(C(c1cccs1)SC)=O)C Cc1cc(F)cc(C)c1C(N1CC2C(CNC(=O)CCN3CCCCC3)C2C1)=O C=CC1OCCCC1C(=O)N(C1(CNC(=O)CCc2csc(=N)[nH]2)CC1)CC C(=O)(CCOCC(C)C)N(CC(=O)N(CC(C)OC)C)CC#C N1(C(CC(=C)Br)=O)CCN(C(=O)CCC(C)(C)[N+](=O)[O-])C2CCCCC12 C(=O)(C(CNC(=O)Cn1cccnc1=O)C(C)C)N(CC)CC1(O)CCC1 C=C(C)C(CC(=O)N(C(C)CNC(c1coc(CCC)n1)=O)C)OCC N1(C(C(C)CN(C)C)=O)CCC(NC(=O)C=Cc2cncn2C)C1(C)C C1(C(=O)NC2CC(NC(C3(F)CCCCCC3)=O)C2)CCC2C(C1)C2(F)F CC(C)CC(F)(F)C(=O)N1CCN(C(C2(C#N)CCOCC2)=O)CC1C CC(C)(C)CCC(F)C(=O)NC1CN(C(=O)CSC(F)F)CC1C1CC1 Cc1cnn2cc(C(N3CC4CC(NC(=O)C(C5CC5)C5CC5)C3C4)=O)cnc12 C1(CC#C)(C(=O)NCC2CC(NC(C3(C4CCCO4)CC3)=O)C2)CCCO1 S(=O)(=O)(c1cccc2c1COC2=O)Nc1ccc2cc(C)c(Br)n2c1 c1(NC)ncccc1C(=O)NC1CC(CNC(C2CC(CC(F)(F)F)C2)=O)C1 C(=O)(C1=CCCC1(C)C)N(CC(C)O)CCNC(C(=Cc1ccccc1)OC)=O CCCC(CC(C)C)C(=O)N1CCCC(O)(Cn2cc(C(O)C(C)C)nn2)CC1 n1(Cc2cn(CC3N(C(C4CC(O)(CC)C4)=O)CCC=C3)nn2)ccccc1=O c1(C(C)NC(=O)COC2CN(C(=O)Cn3ccnn3)C2)ccnn1C C1(C(N2CCC(NC(COc3ccn(C)n3)=O)C2)=O)CCc2nnnn2C1 Cc1ccccc1CCC(=O)NCC1(NC(c2cc(O)ncn2)=O)CCCC1 C(CN=C(NCc1cc(C(C)C)sn1)N(C)Cc1ncnn1C)OCC C12(NC(C(NOC)=O)=O)CCC(C(=O)Nc3cccc(Cl)c3)(CC1)C2 C12(NC(C(CSC)OC)=O)CN(C(=O)CC(C)C)CC1CS(=O)(=O)C2 C1(C(=O)NCc2c(C)scn2)CCN(C(=O)CC(C)(C)O)C12CCC2 CC(C)(C)CN=C(NC1CC(c2cccc(F)c2)C1)N1CC(=O)N(C2CC2)C1 C=CC1(NC(=O)CCC2(NC(c3cccnc3S)=O)CCC2)CCOCC1 Cc1[nH]c2ccc(Cl)cc2c1C(N1CC(CC(=O)O)C(C)C1)Cn1nnnc1C c1(C(=O)NCC(CC=C)NC(=O)C=CC2CCCO2)ccc(C)c(C)c1 c1(C(=O)Nc2scc(COC)n2)cc(I)ccc1[N+](=O)[O-] C1(CC)C(NC(C2CCCN2C)=O)CCCN1C(c1cccc(=O)o1)=O c1(C(=O)NCC2CCC(C)CN2C(c2cccc(Cl)c2)=O)cccn2nncc12 c1(C(=O)NC2CN(C(C3C(C)(CC)C3)=O)C2)ccc2cnccc2c1 Clc1cccc(-c2nc(NCc3cc(Cl)c(Cl)[nH]3)n[nH]2)c1 C(N=c1[nH]c2ccc(F)cc2s1)C1C(NC(C2CCCN(C)C2)=O)CCC1 c1(C(=O)NC2C(NC(CN(CCOC)C)=O)C2)cnc([N+](=O)[O-])n1C C(=O)(CC(C)CC(=O)OC)NC1CC=C(C(=O)NCCC(CCC)C2CC2)C1 Fc1cc(-c2ccc(Cl)cc2)ccc1OCC(F)(F)F.N12CCCCC1C2 N1(C(C2C(CCC)C2)=O)CC(NC(C2COC(=O)C2)=O)C(c2ccnn2C)C1 C1(CNC(C(C2CC=CCC2)NC(C(C)=CC(C)(C)C)=O)=O)CC2(CCC2)C1 C1(CC)CCC(C(=O)N(CC(=O)NCc2cc(C)[nH]n2)C2CCC2)O1 c1(C(C)(C)C)ccc(N)c(C(N2CCC(CNC(C3C4CCN3CC4)=O)C2)=O)c1 Cc1cc(=O)c(C(N2CCCC(CNC(C3(C)CCCCC3)=O)CC2)=O)cn1C c1(C(N(C2CCN(C(=O)CC3C=CCC3)CC2)CC#C)=O)cc(CO)n(C)n1 N1(C(c2[nH]cc(C)c2)=O)CCOCC1CCNC(c1cccnc1C(F)(F)F)=O C1(NC(c2cc(C(F)(F)F)ns2)=O)CCC(NC(C2(C(F)(F)F)CC=CC2)=O)C1 C1(C(=O)NCCN(C(C)C)C(c2csc(C(F)(F)F)c2)=O)C2CCCOC12 CCC(C(=O)NCC1Cn2c(C)nnc2CN1C(C)=O)C(C)(C)CC c1(C(=O)NCC(CC)(C)NC(=O)CNC(c2ccco2)=O)nc(C)n(C)c1C Cc1cc(=N)[nH]cc1C(=O)NC(C)(C)CNC(c1cc(Cl)cnc1C)=O Cc1ccc(CC(=O)NC2CC(C)N(C(=O)CCOC3CC3)C2)cc1[N+](=O)[O-] c1(C(N(C2CN(C(=O)CN3CCOCC3)C2)C)=O)cc(Cl)ccc1[N+](=O)[O-] C1(CO)CCCCC1NCc1cnn(Cc2ccccc2)c1Cl CON1CCC(CC(=O)NCCCCN(C(=O)Cc2csc3nccn23)C)CC1 Cc1cc(CCC(=O)N2CC(CNC(=O)C(C(C)C)c3cccnc3)C2)c(C)s1 N1(C(C2(C)CC(C)(C)C2)=O)CCCC(C2CCCN(C(=O)CSC(=N)N)C2)C1 c1(CC)c(OC)cccc1C(=O)N(CC(CC)NC(c1ccnc(S)c1)=O)C C(CCC(O)C(=O)OCC1CC(C)(C)OC1C)c1cccc(C)c1 C(=O)(CCC#Cc1ccccc1)NC1(CNC(C2C(C=C)OCCC2)=O)CC1 n1(CC)nc(C)cc1NC(C1CN(C(=O)CCc2ncccc2C)CCN1)=O C(=O)(CCC(C)N(C)C)N(CCC(c1cccs1)NC(C=CC(C)C)=O)C c1(C(=O)NC(C2CN(C(Cc3nc(C)[nH]n3)=O)C2)C)cc(C(C)C)oc1C C1(NC(CSCC)=O)C2CC3CN(C(c4ccc(=O)n(CCF)n4)=O)C1C3C2 c1(-c2ncc(C(=O)NCC3C(CNC(C(CSC)O)=O)C3)s2)ccccc1F CC1(C)C(=O)CC1C(=O)NC(C(N1CCC(c2nn[nH]n2)C1)=O)c1ccco1 C(CCCCC(=O)NCCC1CN(C(=O)CC2CC3(CC3)C2)CCCO1)=CC c1(OC)c(Cl)cc(C(=O)NC(C)CCNC(c2cnc(=N)[nH]c2)=O)nc1Cl c1(C(=O)NCC2N(C(C3(C)CC(C)OCC3)=O)CC2)ccc2c(c1)C(C)C(C)O2 S(=O)(=O)(c1ccccc1)NCCC(N1CCC(NC(=O)CC2C=CCC2)CC1)=O C1(NC(C2(S(N)(=O)=O)CC2)=O)C2CC3CN(Cc4ccnc5[nH]cnc45)C1C3C2 C(=O)(CCC(F)(F)C(F)F)N(CC(CC)NC(c1cncc(N(C)C)c1)=O)C c1(C(N(C(C(=O)NCCCC2CCOCC2)C2CC2)C)=O)c[nH]c(C(N)=O)c1 Cc1c(C(=O)NC2CC(NC(c3ccon3)=O)C(O)C2)sc2ccsc12 Cc1c(C(N2CCCC(N(C(=O)CC(C)F)CCF)C2)=O)sc2cccc(F)c12 C1(C(N(C(CC)C(=O)N(C2CCN(C)C2)C)C)=O)CC(N=[N+]=[N-])C1 Brc1ccc(-c2cn(CC3CC3)nn2)cc1.C12N(CC1(C)C)C2 c1(C(=O)NCC(CNC(c2occc2C)=O)OC)csc(C(F)(F)F)n1 n1(CC(N2CCN(C(c3nc(CC)oc3)=O)C3C2C3)=O)cc(C)c(O)nc1=O C1(OC)CC2(C1)CC(C(=O)NCC1(C)CCN(C(=O)C(O)c3ccsc3)CC1)C2 c1(CC(N2CCC(O)(CNC(CNS(NC)(=O)=O)=O)C2)=O)cnc2n1CCOC2 C1(NC(C(C)=C2CCCC2)=O)CCCC(CNC(c2ncn(C(C)(C)C)n2)=O)C1 N1(C(=O)OC(C)(C)C)CCC(C)(C(N2C3CN(C(=O)CN)CC23)=O)C1 c1(NC(C(C2CCOC2)NC(c2cc(CC)[nH]n2)=O)=O)ccc(CCO)cc1 C1(C(N(CC=C)CCC)=O)CCCN(C(c2cc(Cl)cn2C)=O)CC1 CCCC(C(=O)NCC(c1ccco1)O)NC(=O)C(C)(C)CC1CC1 N1(C(C(C)(C)CC(F)(F)F)=O)CCC2(CO)CN(C(=O)C3=CCCCC3)CC2C1 c1(C(N(CCCN(C(=O)CCCC2CCOCC2)C)C)=O)cc(N)cc(O)n1 S(=O)(=O)(c1cc(C(F)(F)F)cc(Cl)c1)N1CCC(NC(C(=O)N(C)C)=O)C(F)C1 N1(C(Cc2scc(C)c2)=O)CCCC(C2CN(C(=O)CSC3CCOC3=O)C2)C1 C1(CC(=O)NCCOC2(C)CCC2)CCCCN1C(C1CC=CCC1)=O Cc1cc(N2CCC(c3nc(C)cs3)C2)nc(=NCCC2SCCS2)[nH]1 c1(OC)cc(C(N2CCCCC(NC(C3CC3OC)=O)C2)=O)ccc1OC(C)C c1(CC(C(=O)N(C)Cc2nncs2)NC(=O)CNC(N)=O)cnn(C)c1O c1(C(C(=O)Nc2cncn2C)NC(C2CCN(C(C)=O)C2)=O)c(C)cccc1Br c1(CC)cc(C(=O)NC(CNC(=O)Cc2csc(C(F)(F)F)n2)C(C)C)nn1C c1(OCCC(N2CCC(CNC(C=CCOC)=O)(CO)C2)=O)cc(C)cc(C)c1 S(=O)(=O)(c1cccc2nonc12)N1CC(C(c2nnc(-c3ccco3)o2)CC)C1 c1(C(N(CC(=O)NCC2(O)CCOCC2)CC#C)=O)cc(C)nc(C)c1 n1(CC)cnc(C(=O)NC(C2CCCC2)CNC(C2(c3ccn(C)n3)CC2)=O)n1 C(=O)(NNc1cccc(C(F)C(F)(F)F)n1)c1c(F)ccc(C(N)=O)n1 C1(C(N2CCC(OC)C2(C)C)=O)CCN(C(C2CCC3(CCC3)C2)=O)C(C)(C)C1 c1(OC)ccnc(OC)c1C(=O)NC(C)C(C(C)C)NC(c1ccccc1O)=O CCCCCCC(F)C(=O)N1CCN(C(c2cnn(CCO)c2)=O)CC1CO c1(C(N2CCC(C)(NC(c3cccc(OC)c3)=O)C2)=O)cc2c(O)cccc2[nH]1 C12(CNC(c3ccc(CC)cn3)=O)CC(NC(=O)C(N)=O)(CCO1)C2 c1(CN2C(C(N3CCC(C(C)(C)O)C3)=O)COCC2)cn2cccnc2n1 c1(OC)ccnc(F)c1C(N1CCC(O)C(NC(c2cc(F)ccc2F)=O)C1)=O C(=O)(C1=CC2C=CC(C1)C2)NC(C1(O)CCN(C(=O)CCc2ccncn2)C1)C C1(C(N(C)CC2(O)CN(C(=O)CC(C)(F)F)C2)=O)CC2(CCC2)CO1 C(C)(C)(CC(=O)Nc1ccc(Cl)nc1)N(C)C(C1CC1C(F)F)=O CN1CCCCCC1C(=O)NC1(CF)CCN(C(=O)CCc2cnc[nH]2)C1 Cc1cnccc1C(=O)NC1CCCC(NC(c2cnsn2)=O)C1 CCC(CO)(C(=O)NC1CC(CNC(c2cscn2)=O)C1)OC CCC(CC(=O)N1CCC(N(C(=O)CCc2nc(CC)no2)CC)C1)C1CC1 N1(C(C2CCCC2(C)C)C(=O)NCCSC)CCS(=O)(=O)C2CCCCC12 C(=O)(C1SCCc2sccc21)N(CCCCNC(=O)CCOC1CCCOC1)C c1(C(C(=O)NCc2cccc(F)c2F)N(C(C)CC#N)C)cccn2ccnc12 c1(C(N2CC(CC(=O)Nc3c(OC)nn(C)c3)(OC)C2)=O)cccc(C)c1F C1(C(=O)NC(c2ccc(F)cc2)CNC(CP(C)(C)=O)=O)OCC2COCCC12 c1(C(N2CC(NC(C3(Cl)CC34CCC4)=O)C(F)C2)=O)ccc([N+](=O)[O-])c(O)c1 N1(C(C(COC)NC(C)=O)=O)CCC2(CCN(C(=O)Cc3cnnn3C)CC2)C1 N1(C(C(c2c(C)cccn2)(F)F)=O)CCCN(C(=O)CC23CCC(CC2)C3)CC1 C1(C(N2CC3C(CNC(=O)COC4CCOC4)(C3)C2)=O)CCC2(CCCCC2)C1 C1(CNC(c2cc(C)no2)=O)(NC(c2cc(=O)n(C)o2)=O)CCCCC1C CCC(C(C)CN(C)C)NC(=O)C(CC1CC1)NC(=O)CN=[N+]=[N-] C(CCCN=c1nc(C(C)(C)C)[nH]s1)NC(c1cc(OC)nc(C)c1)=O c1(OC)cc(N2CC3(CC(NC(c4ccc(C)c(C)n4)=O)C3)C2)nc(OC)n1 CCC(CC(=O)NC(C1CCN(C(c2nc(C)nn2C)=O)CC1)(C)C)OC C(CCC)(C(=O)NC12CC(NC(=O)C(C3CC3)OC)(C1)C2)=CCC N1(C(Cn2c(C)nnn2)=O)CCCN(C(c2scnc2C(C)C)=O)CC1CO c1(C(=O)NC2CCC(C)(CNC(c3c(C)nc(C)s3)=O)C2)c(C)oc(C)c1C c1(CCC(C)(c2nnnn2C2CC2)NCC(C2CCOC2)OCC)ccc(F)cc1 c1(OC2CCN(C(C(C3CCOC3)OCC)=O)CC2)cccc(C#N)c1 C1(C(N2CC(O)(CNC(=O)COC3CCCC3)C2)=O)C2CCC(C2)S1(=O)=O c1(C(N2CCC(C(C)NC(c3n(CC=C)ccc3)=O)C2)=O)sc(=NCC)[nH]c1C C1(CC(=O)NC2CN(C(C3(CC=C)CCOC3)=O)C2)CCOCC1OC N1(C(C2CC(OC)C2)=O)CCC2(CCC2NC(C2CCC(=O)O2)=O)CC1 N1(C(CN(CC)CC)=O)CCC(CNC(c2occ3c2CCC3)=O)C(F)(F)CC1 Cc1cc(C(N2CC3CC(NC(C4CCCC4(C)C)=O)C3C2)=O)cc([N+](=O)[O-])c1 C=C(C)CCCNC(=O)C(C)=CCNC(c1cc(C)sn1)=O C1(CCC)CN(C(c2cnn(C)c2Cl)=O)CCN1C(c1nc(C2CC2)cs1)=O C(C)(N=c1[nH]ncs1)C1OCCN(C(c2ccc(OCC)nc2)=O)C1 c1(C(=O)NC2C(NC(c3cn(CCCC)nn3)=O)CC2)cn(C)c2ncccc12 C1(CC(=O)N(C2CC3(CNC3)C2)CC2CC2)CCC2CNCCC2C1 c1(C(C)OC)nc(C)c(C(=O)NCC2(F)CN(C(=O)Cc3cncc(C)c3)C2)s1 c1(CC)ccccc1C(CNC(C1CC1C#N)=O)NC(=O)CNc1nccs1 C1(CCNC(C(C)Nc2scc(C)n2)=O)CN(C(=O)Cc2cnc(C)s2)CCO1 N1(C(CSC(C)C)=O)CCOC(CC(N2CCC(C)(C(C)C)C2)=O)C1 c1(C(F)(F)F)cccc(CNC2(C3CCC3)COC2)c1 C1(NC(c2cc(C)cc(O)n2)=O)CC2CCC1CC2NC(C1(C)C=CCC1)=O C1(NC(c2cc(C)no2)=O)CCC(NC(C2CC2(c2ccccc2F)C)=O)CC1 c1(C(N2C3CN(C(Cc4cc(OC)ncc4)=O)CC32)=O)cc(Br)ncc1[N+](=O)[O-] Cc1ncc2ccccc2c1C(=O)NCC(C)NC(=O)Cc1scnc1C C(=O)(C(C)(C)CC(=O)N1CCSCC1CCNC(=O)C(C)c1cc[nH]n1)OCC C(=O)(C(C)CC(C)(C)C)NC1CN(C(C(CC)CC)=O)CC(C)C1 c1(-n2cc(C3CCN(C(C4CNC(=O)N4)=O)C3)nn2)cccnc1Cl c1(C(N2C3CCC2CN(C(C24CCCC2OCC4)=O)C3)=O)cccc2nonc12 c1(OC)cccc(C(N2CCC(F)C(NC(=O)CNC(C)=O)C2)=O)c1F C1(CC=C)(C(=O)NCCCOCCCO)CCCN1C(c1cc(C)ncn1)=O c1(C(=O)NC(C)CNC(C2CCS(=O)(=O)C2)=O)c(O)c2ccccc2n(C)c1=O Cc1ccccc1C(C)N(C)CCOCC(F)(F)F.C1(N)COC2(CCC2)C1 C(=O)(CCCCC(=O)NC1CCN(Cc2csc(C)n2)CC1(C)C)OC c1(N2C(CCCNC(C3CC(O)(CC#C)C3)=O)CCC2)cncc(C#N)n1 S(=O)(=O)(c1ccc(C(=O)NC(c2ccc(F)c(F)c2)C)cc1)N(CC=C)C C1(N(C)C(=O)NCC2(c3cccs3)CC2)CCC(F)(F)CC1 c1(C(N(C2CN(C(C(C)C(C)(C)C)=O)C2)C)=O)ccc2nnn(C)c2c1 C1(O)(CCn2cc(CSC)nn2)CCN(C(=O)CC(C)C2CC2)C1 C1(C(=O)NC)(CF)CCN(CC2CC2Br)C1 S(=O)(=O)(c1ccc(C#N)c(NCCC(C)P(C)(C)=O)c1)NCCN(C(C)C)C1CC1 N1(C(C(=O)N(C)Cc2cc(-c3ccc(F)cc3)nn2C)=O)CCCNC(=O)CC1 c1(C(=O)NCCC(C)NC(c2cncc(C(F)(F)F)c2)=O)cc2c(ccn2C)s1 CC(CNC(C1C2CN(C(c3cccc(Cl)c3)=O)CC12)=O)S(C)(=O)=O c1(SC)ccc(OCC(N2CCC(C(C)NC(C3CCCC3)=O)C2)=O)cc1 C1(CCC(=O)OCC)C(=O)N1.CCC#CCCNC(C)(C)C c1(COCC)nc(N2CCC(CNC(=O)C(C)C3CCC3)C2)cc(Cl)n1 c1(OCC(=O)NCC(C(CC)C)=O)cc([N+](=O)[O-])ccc1F N1(C(c2cocc2Br)C(=O)NCCSC)CC(C)OC2(CCC2)C1 N1(C(c2cc(C)n(C(C)C)c2)=O)CCN(C(=O)CN2CCCC2C)C(C(C)C)C1 Cc1oc(Cl)nc1C(=O)NCCC1CCN(C(=O)CC(C)n2ccnc2)C1 N1(C(C2(OC)CCOCC2)=O)CCN(C(=O)C2=CCC2)CC12CCC2 C1(C(=O)NCC(CN(C(Cc2cnc(C)[nH]2)=O)C)(C)C)CCn2c(cnc2C)C1 Cc1cnc(C)c(N2CCN(C(=O)NC3CC(=O)N(C(C)C)C3)CC2)n1 C1(C(N2CC(CNC(c3c(CC)onc3)=O)OCC2)=O)CC2(CC(=O)C2)C1 CN1CCCC(NC(C2CN(C(c3ccccc3C#N)=O)CC2(F)F)=O)CC1 C12(C(=O)NCC=CC(=O)NCC(C)SC)CC(F)(C1)C2 N1(C(Cn2nc(C)oc2=O)=O)CCC(CO)(CNC(C2CC=CCC2)=O)CC1 C1(NC(=O)CCC2CCOC2)CCN(C(=O)C=CCOCc2ccncc2)CC1 c1(N(CC(=O)NC)C)nc(N(CC(C)OC)C)nc2cccc(F)c12 Cc1cc(CNC(=O)Cc2cnsc2)oc1C(=O)NCCN1CCCC(O)C1 C(=O)(C(CCc1ccco1)N1CCOC(CCc2ccccc2)C1)NC1(C)CC1 c1(OC)cc(C(N2CC(CC(C)C(N(c3ccc[nH]3)C3CC3)=O)C2)=O)cc(F)n1 N1(C(c2cc(C)nc(O)c2)=O)Cc2n[nH]cc2C1C(=O)N1CCCC(C#N)C1 n1(CC(=O)NCCC(CNC(CCC(=C)C)=O)O)nc(C(F)F)c2c1CCC2 N1(C(C2C(C)CC(=O)NC2)=O)CCCC(C2CN(C(=O)CC3C=CCC3)C2)C1 C12(NC(c3c(O)cccc3Cl)=O)CCC(CC1)N(C(=O)CCC1CCCOC1)C2 c1(C(N2CCCN(C(CC3(C)CC3F)=O)CC2)=O)cc(F)c(Br)c(Cl)c1 C1(C2CC2)(C(=O)NCCC2CCN(C(=O)C=Cc3nccs3)C2)CCC1 C1(CNC(c2nn(C)c(Cl)c2)=O)CN(C(C2SC3C=CC2CC3)=O)CCCO1 N1(C(=O)C(F)(F)Cl)C(C(N2CCC3(CCOC3)C2)=O)CC2CCCCC12 C1(C(=O)NCC(CC)(CC)NC(C2N(CC)CCC2)=O)COCCN1C=O C1(C(=O)NCc2cc(C(N3C(C)(C(=O)NC)CC3)=O)on2)CC(=O)C1(C)C C(=O)(C(CC(C)C)ONC(C12CCC(CC1=O)C2)=O)NC(CCC)C(=O)NC CC(C)C(C(=O)NC(C)CNC(c1c[nH]nc1C(C)(F)F)=O)n1cncn1 C(c1ccc(C#N)cc1)=CC(=O)NC1CCC(C)N(C(c2cncnc2)=O)C1 CCC(CCC(=O)NC(Cc1cn[nH]c1)C(=O)NCC1(O)CCC(C)C1)OC C1(OC)CN(C(C2(OC)CC2)=O)CC1C(N1CC(C)(O)C1)=O C1(C)(C(=O)NC2C(SC)CN(C(=O)CC3(O)CCC3)C2)CC(=O)N(C)C1 C1(C(=O)NC2CC(F)(CNC(c3cnc(C(F)F)nc3)=O)C2)CCS(=O)(=O)C1 CC(C)CC(O)CC(=O)N1CCC(C(=O)NC2(C)CC(O)C2)C12CCC2 C1(C)(C(=O)NCC(C)NC(c2ncccc2C(F)(F)F)=O)CCCOC1 C12(C(=O)OC)COC(C(N3CCCCC3CNC(=O)CCCSC)=O)(C1)C2 N1(C(C(=O)NCCOCCO)=O)CCCC(c2nnc(S)n2C2CC2)C1 C=CCC(C(=O)N1CC(OCC(=O)NCCC23CCCC2C3)C1)OC C1(CCCC)CCC(NC(C2(NC(=O)OC(C)(C)C)CC(CO)C2)=O)C1 Cc1ncc(C(=O)N(C2CCN(C(c3csc(Br)c3)=O)C2)C)c(=N)[nH]1 N1(C(C(CC)c2ccccc2)=O)CCN(C(=O)C=C2CCN(C)C2)CCC1C C(=O)(C(F)(F)CO)NC1C(CNC(CNS(CCOCC)(=O)=O)=O)COC1 C=CC1(CC(=O)NCC2CCN(C(=O)Cc3ccoc3)CC2CC)CCOCC1 C(N=c1cc(Cl)nc(C2CC2)[nH]1)C1C2N(C(Cn3nnc(C)n3)=O)CC(CC2)C1 C1(NC(C=CC)=O)CN(C(C2CC3(C2)CC3F)=O)CC1N=[N+]=[N-] N1(C(CCOCCNC(c2ccncn2)=O)=O)CC2CC1C(F)(F)C2 N1(C(c2c(C)cc(CO)o2)=O)CCC(CNC(=O)CCN2CCOC2=O)C(C)C1 c1(C(N(CCCN(C(C(C)(C)OCC)=O)C)C)=O)nc(C)ncc1Cl C=CC1(C(N2CC(C)(F)C2)=O)CCN(C(=O)COc2ccsc2)CC1 C1(O)(CC(N2CCC(CNC(C(C)CO)=O)C2)=O)CCCCC1 c1(C(=O)NCCC2CN(C(CN(C(C(C)C)=O)C)=O)C2)c(C(F)F)cccc1F C1(N(C(c2scc(COC)c2)=O)C)CCCN(C(=O)C(COC(C)C)OC)CC1 c1(NC2CC3CC(NCC4C(C)(C)S(=O)(=O)CC4)C3C2)c(Br)cccc1[N+](=O)[O-] c1(CC)cnc(Cl)nc1N1CCCC(C)(NC(c2sccc2Cl)=O)C1 C1(C(=O)NC2CC(OC)C(O)C2)CCCCC(C)(C)C1 c1(C(=O)NCC(N(C)C(c2ncc(Cl)nc2Cl)=O)C2CC2)cccc2c1OCC2 C=CCC(CC(=O)NC1CCCCCC1F)NC(=O)CC(=O)OC N1(C(C)C)CCC(NC(C2CCN(C(=O)CCN(C)C(C)=O)C2)=O)CC1 C1(CNC(C(CCSC)O)=O)CN(C(=O)C(C)(C)n2cnnn2)CCC12CCC2 C1(NC(c2cnn(C)c2)C)CCN(C(=O)OCC)CC1C.C(C)(C)(C)O N1(C(c2cncc(C=C)c2)=O)CCN(C(C2CCN(CC)C2)=O)C2CCC12 c1(C(C)(C)C)ncc(S(=O)(=O)N2CCOCC2Cc2nn[nH]n2)o1 N1(C(c2c(C)oc(Cl)n2)=O)CCC2(C1)CN(C(=O)Cc1cncc(C#N)c1)C2 N1(C(c2nn(C)c(Cl)c2Br)=O)CCC(CNC(c2cc[nH]n2)=O)C12CCC2 Cc1cccc(C)c1OC(CNCc1cccc(NC(=O)OC(C)(C)C)n1)=O c1(C(=O)NC)ccc(-n2nc(-c3cccs3)nc2CCN2CCCCC2)cc1 Cc1cc(C#N)cnc1C(=O)NCCCN(C(=O)CC1CS(=O)(=O)CCN1C)C CCCCCCCC(F)C(=O)NCC1CN(C(c2ccc(C)c(C)c2)=O)CC1C N1(C(CCC)=O)C(C)CC2CN(C(C3CCCC3(C)C)=O)CC12 N1(C(c2cnc(COC)nc2O)=O)CCN(C(c2csnn2)=O)CC(C)(C)C1 C(=O)(CCC(=O)NCC1CCN(C(=O)Cc2csnn2)C1)N(C(C)C)C c1(C(=O)NC2CC(F)(CNC(CC3(OC)CC3)=O)C2)cc(Cl)cc2ccncc12 c1(C(=O)NC2CN(C(C(=O)NCC)=O)CC(O)C2)ccc2nsnc2c1 c1(C(N(C2CN(C(C3(C)ON=C(C(C)C)C3)=O)C2)C)=O)cc2c(=O)[nH]ccn2n1 N1(C(c2c(F)ccc(OC)c2)=O)CC(C2CCCN(C(=O)CC34CC(C3)C4)C2)C1 C#CCC(CC(F)F)C(=O)N(CC(=O)NCC1CCN1CC)CCC C1(CNC(C2(CC)CC2)=O)CC(NC(=O)Cn2ccc(C)n2)C1(C)C Cc1c(Cl)c(C(=O)NC2CN(C(=O)CC3CCC=CCC3)CC2C)nn1C C1(NC(CN(CCC#C)C)=O)CC2(C1)CC2NC(=O)C=CC(=O)N(C)C Cc1cc(C)c(C(=O)NC2CCC3(C2)CN(c2ncncc2I)C3)cc1C C(=O)(C(C)(C)C(C)(C)O)N1CCC(OC)(CNC(=O)CCc2cnn[nH]2)C1 C(C(C(=O)N(C(C)C(=O)NCC1CCOC1C)C)OC)OC N1(C(C2C(C)CCOC2)=O)CCC(CC(=O)NCC2(CC(N)=O)CC2)C1(C)C Cc1nc2[nH]c(C(=O)NCC(O)CNC(c3ccc(CF)cc3)=O)cc2s1 C1(NC(c2ccc(OC)s2)=O)CC2(C1)CC(CNC(C1(C)CS(=O)(=O)C1)=O)C2 C(=O)(CS(=O)c1ccc(Cl)cc1)NCC1(O)CN(C(Cc2n(C)ncc2)=O)C1 c1(OCC)cccc(CCC(=O)NC(C)CNC(C2CC(F)(CF)C2)=O)c1.C1CC1 c1(OCCCC)cc(OC)ccc1C(=O)NC1CC1NC(=O)C(O)CC(N)=O CC1(C)COC(CC(N2CC(C3(NC(C4CCS4(=O)=O)=O)CC3)C2)=O)CO1 N1(C(C(C)NC(CC)(C)C)=O)CCCCC(C(=O)N(C)Cc2cnn(C)c2)C1 c1(C(N(C(CNC)CO)CC)=O)nc(C)ccc1NC1(O)CCCOC1 C(=O)(CCCC(=O)NCC1(F)CCN(C(=O)C(F)n2ccnc2)C1)N(C)C c1(C(=O)NCC(C)NC(c2ccc3c(c2)COC3)=O)cc(Cl)c2[nH]c(O)nc2c1 N1(C(C=Cc2n(CC)ccn2)=O)CC(NC(=O)COC)CC(C)C1 N1(C(=O)CCN2CCC(O)CC2)CC2CC1CN2C(C12CCC(O)C1CC2)=O CCCCC(CC)CC(=O)NCC(C)(C)OCC(=O)N(CC)Cc1cn[nH]c1 CCC(F)(F)C(C)(C)C(=O)NCC1CN(C(=O)CCOC(C)C)CCO1 CC(O)C(F)(F)C(=O)N1CCCC(CCC(=O)N(C2CCCC2C)C)C1 CC1(C)C2CCC1(c1nc(-c3cccc(F)c3O)no1)C2 c1(C(CC)C)nc(C2CCCCC2O)n(CCc2ccccc2)n1 CC(C(=O)NC1CC(C(N2CC(F)(F)CC2C)=O)CC1O)C(C)(C)C c1(NC(=O)NC(c2nc(CC)[nH]n2)C)cc(Cl)c(Cl)cc1Cl c1(C(=O)NCCNC(C(C)C)=O)n[nH]c2c1CN(C(=O)C=CC1CCOCC1)C2 C1(NC(=O)Cc2cnns2)CCC2(CCCN2C(C2C3CCCCCC23)=O)CC1 c1(C(N(C)CC2CCCN(C(=O)CC3(CO)CC3)C2)=O)cnn2c(=O)cc[nH]c12 CN1CCC(C(=O)NC2(CNC(=O)CC3CCN(CC(F)(F)F)C3)CC2)C1 c1(-c2cccc(CC)c2)cccc2[nH]nc(C(=O)NCc3cccc(F)c3)c12 N1(C(c2cc(C)nn2C2CC2)=O)CCCC2(CCN(C(C3(C)CC(C)C3)=O)C2)C1 C1(NC(c2ccc(SCC)nc2)=O)CCN(c2nc(Cl)ncc2F)CC1(C)C CCCCS(=O)(=O)CC(=O)N1CCOCC1CNC(C1COCC(C)(C)O1)=O C1(NC(C(CC#C)C)=O)CC2C1CCN2C(=O)Cc1ccc(Br)cc1OC c12ccc([N+](=O)[O-])cc1N2.c1(OC)cc(NC(=O)C(C)(C)C)c(C(=O)O)cc1F N1(C(C2(CC=C)CN(C(=O)C(F)OC(F)(F)F)C2)=O)CCN(C)CC1C C12(C(=O)NC(C=C)CO)CCCC1CN(C(c1cc(O)ncc1F)=O)C2 c1(C(=O)NC2(CC=C)CN(C(C3(C(=O)NC)CC3)=O)C2)c(Cl)ccnc1C C(=O)(CC(C)(C)Cc1nn[nH]n1)N(C1CCN(C(c2ccc(C#N)cn2)=O)C1)CC c1(CC)ncc(-c2cn(CC3(CNC(=O)C(c4ccco4)C)CC3)nn2)o1 C1(CNC(C2(CC=C)CC2)=O)CN(C(=O)CCSCC(C)C)CC(C)(C)O1 C1(C(=O)NC(CNC(C(c2cccnc2)C)=O)(C)C)CCCCN1C(N)=O N1(C(C(CC=C)OC)=O)CCN(C(c2ccncc2Cl)=O)C2CC12 C1(C(N2C3C(NC(C=CC(C)(C)SC)=O)C(CC3)C2)=O)CCCC1P(C)(C)=O N1(C(CCc2c(C)ncs2)=O)CC(CO)C2(C1)CN(C(=O)C(C)C(F)F)C2 c1(C(=O)NCc2cn(CC)nc2)ccc(OCC2CCCCO2)cc1C C1(CC)(NC(C2CC(C)(O)C2)=O)CCN(C(C2CCN(C)C(=O)C2)=O)CC1 CC(C)CC(C)(CNC(C1(C2CC2)CC1)=O)NC(=O)C1=CCSC1 c1(N(C)Cc2c(CC)cccc2)nc(NC(C)C(C)CO)c2ncsc2n1 c1(OCCSC2(C#C)COC2)c(C)cc(C#N)cc1C c1(OCCC(=O)NCC23N(C(CCC)=O)CC(C2)C3)cccc2ccccc12 C1(O)(CNC(CC(=C)C)=O)CCCN(C(=O)C(C)Cc2ccco2)C1 n1(CC)nc(C2CC2)cc1C(N1CCCC1(C)CNC(c1c[nH]nc1OC)=O)=O C(=O)(C(C)CC=Cc1cccs1)NC1(C#C)CCC1 N1(C(C2N(C(c3c(C)snc3)=O)CCSC2)=O)Cc2ncsc2C1 CC(N=c1nc2scnc2c(NC(C)CN2CCCCC2)[nH]1)c1ccc[nH]1 CC1(C(=O)NCC2CCCCO2)CCN1C(c1n[nH]cc1Cl)=O C(CCCCC(=O)NC1CC(CCC(=O)NCC2CC(C)(O)C2)C1)OCC C1(NC(c2n(CC)nnn2)c2noc(C)n2)CCC2CC1CO2 CC1OCCC1(C)C(=O)NCC(C)(C)NC(c1cc(OC2CCCC2)ncn1)=O c1(C(N2C(C3CCN(C(c4cc(C)c(C)o4)=O)C3)CCC2)=O)cccc(F)c1N C12(COC(c3cc(C(C)C)nn3C)=O)CC(C)(C1)C(CO)O2 C=C(C)CC(C(=O)NCC1CCCCN1C)NC(=O)C(=O)C(C)(C)C CCC(CC(=O)NC1CC(NC(=O)CC(C)C(=O)OC)C1)C(=O)OC(C)(C)C c1(C(=O)NCC2(F)CC(CNC(=O)CO)C2)cncc(-c2ccc(Cl)cc2)c1 CC(O)(CC(=O)NC1(CNC(C2CCCC2O)=O)CC1)C1CC1 C(CN=c1[nH]nc(-c2ccccc2)s1)N(C(c1cnoc1C)=O)CC N1(C(C(CC)OCC)=O)CC2CN(C(=O)C=C(C)C(F)F)CC2C1 O=C(CCCC(F)(F)F)NCC1CC(F)CN1C(=O)C=CCN1CCOCC1 c1(C(=O)NCCC2N(C(CC3(C#N)CC3)=O)CCSC2)cccc2nonc12 C1(NC(c2cn(CC=C)nn2)=O)CC(C(=O)NCCC2C=CCC2)CC1O Cc1c(N)ccc(C(=O)NC(C2CCN(C(=O)C(C)CC(F)(F)F)C2)(C)C)c1F c1(OC)cc(NC(C)CNC(=O)Cn2cnc(C(N)=O)n2)nc(OC)n1 C1(NC(C2C(C)(Br)C2)=O)CCN(C(=O)C=CC2CCCCCC2)C1(C)C C(=O)(C(COC)CC(C)C)NCCN(C(c1c(C)nnn1CC)=O)CC C(F)(c1ccccc1)=CC(N1CCC(CCNC(c2ccc(F)cn2)=O)CC1)=O CC1CCC2(CCN(C(=O)C#CCNC(c3nccnc3C(N)=O)=O)C2)C1 CC1(CNC(=O)C(O)Cc2cnc[nH]2)CCCN1C(C1CCC(C(N)=O)CC1)=O c1(C(=O)NC2CN(C(C(C=CCCC)O)=O)CC2O)nc(C)ccc1C CC(C)CCOCC(=O)NC(C)CNC(C1CC(OCC2CC2)C1)=O C1(NC(C2(CCOC)CC2)=O)CCN(C(C2CCCCC2C)=O)C(C)C1 C1(NC(C(N2C(C(=O)OC)OCC2)=O)=O)C2CCC(C2)C1c1ccccc1 C1(C(=O)NCC2C(OC)CC2)CCOC1CNC(=O)CCOCC(C)(C)C Cc1ncc(C(=O)N(C(CNC(=O)C(C2CCCO2)C2CC2)C2CC2)C)s1 Cc1nc(O)sc1C(=O)N.c1(C(N2C(C3CCC3)CCC2)=O)ccc(C2CC2)nc1 c1(OC)c(C(N2CCC(CNC(c3ccoc3)=O)C(C)C2)=O)occc1=O N1(C(C(C)NC2CCOC2)=O)CCC(O)C(N(C(=O)C=C(Cl)CCN(C)C)C)C1 N1(C(C2C(CC)C2)=O)CC(O)(CNC(C2CC(C)(C)C2)=O)C1 c1(CC(N2C(CNC(C3CC(O)C(F)C3)=O)CCC2)=O)ccc([N+](=O)[O-])cc1 C1(CNC(CC2(C)CC(F)(F)C2)=O)CCC2(CN(C(c3csc(O)n3)=O)C2)O1 CC1CN(C(CCc2ccccc2)C(=O)Nc2ccc(F)cc2)CC(C)S1=O O=C1C(=O)N(C(=O)c2cccn3c(I)cnc23)c2ccc(F)cc21 N1(C(c2ccc(CNC(CCCC(C)(C)C)=O)cn2)=O)CC2CCC1C(O)C2O CCCCCC(O)CNC(c1ccc(CNC(C2CCC(C)O2)=O)s1)=O c1(C(=O)NC(CNC(C2CN(C(N)=O)C2)=O)C2CC2)cc2c(nn1)CCC2 N1(C(CC)=O)CCC(C(=O)NCCCN(C)C(c2ccc(SC)s2)=O)C1 N1(C(c2c(C#C)c[nH]n2)=O)CCC2(CCN(C(=O)Cc3cc(CC)nn3C)C2)C1 CCC(CC)(CO)C(=O)NCC1C(C)CCN1C(=O)C=Cc1ccco1 CCC(CC)C(C(=O)N(CCCNC(=O)CC1CCOC1)CCO)OC N1(C(CC2C(CNC(C3(C(C)C)CCC3)=O)C2)=O)CCC(C2(C)CC2)C1 c1(C(=O)NCC2(C(=O)Nc3ncc(C(N)=O)nc3)CC2)ccc(Br)c([N+](=O)[O-])c1 C(=O)(C#CC1CCCO1)NCC(CC(C)C)(C)NC(c1cnc(C(C)(C)C)s1)=O C(=O)(C#CC(C)(C)O)NCC(CNC(c1cc(CCC)n(C)n1)=O)(C)OC c1(C(=O)NCCSC2CCN(C(CN(C)CC)=O)C2)ccccc1C(C)=O c1(CN(CCN(C)C)C(c2[nH][nH]c(=N)c2Br)=O)ccc(Cl)c(Br)c1 Cc1cccc(C(F)(F)C(=O)NCC(C2CCCC2)NC(=O)C(C)C2CC2)n1 C1(CNC(CN(CCOC)C)=O)CCC(CNC(=O)C=C(C)c2ccsc2)CC1 CC1=NOC(CCNC(=O)C(O)C2CN(C(C3(Cl)CCC3)=O)C2)C1 N1(C(C2CCN(C(=O)c3c(CC)n(C)nc3)O2)=O)CCc2ccsc2C1 C=CCC(CNC(C1(C)CCN(C)C1)=O)C(=O)NCCC1(C)CCOCC1 c1(CCC(=O)NCC(C(C)C)NC(=O)CNC2CC2)c(F)cccc1Cl C1(NC(C(=O)Nc2cccc(C)c2)=O)CCN(C(=O)CSC2CC2)C12CCC2 N1(C(c2cccc(Br)c2OC)C(=O)NCC)C2CCC1C(C)C(O)C2 c1(C(=O)OC)[nH]nnc1C(=O)NC(CN1CCCCC1)C(C)C N1(C(Cc2n(C)nnc2)=O)CC(NC(c2ccccn2)=O)CC12CCCOC2 Cc1nc(CO)sc1C(=O)NCC1CC(O)CN1C(=O)C(C)n1cnnn1 Cc1ccc(Cl)c(C(=O)NCC2(O)CCS(=O)(=O)C2)c1N C(=O)(C(CC(C)C)NC(=O)C(C)COC)N(C(CC)CO)C c1(C(=O)NCC(CC(C)C)NC(C(c2cc(C)oc2C)C)=O)cn2c(n1)CCC2 c1(CCCC(N2CCC(N(C(C3C(C(C)C)C3)=O)C)C2)=O)ccc(F)cc1 N1(C(c2ccncc2)C)CCOCC(C(=O)NCCSc2ccccc2)C1 C(=O)(CC(C(F)F)NC(=O)C(C)NC(=O)C1CC1)NC(CC=C)C C1(CC)(NC(=O)CC2CCCC(=O)N2)CCN(C(c2cc(F)cnc2O)=O)CC1 c1(C(N(C)CC2CN(C(=O)Cn3ccnn3)C2)=O)[nH]nnc1C1CC1 c1(C(C#C)(C)NC(=O)NCC(C)F)ccccc1 c1(OC)cccc(C(=O)NC2COCC2NC(=O)Cc2ccnnc2O)n1 CN1CCC2(CCN(C(=O)CSCCNC(=O)CC3CCC(C)(C)O3)C2)C1 CCC(CC)(CCC(=O)N1CC(O)CC1CNC(=O)Cn1cc(C)cn1)[N+](=O)[O-] C(=O)(C(C)(O)C(F)(F)F)NCC(c1cccc(C)c1)NC(=O)CCc1nc[nH]n1 c1(C(N2C(CC)CN(c3nc(OC)ncc3F)CC2)=O)ccc2nc(Cl)sc2c1 C(C(CC1CCCC1)C(=O)NCC(C)(C)CCO)NC(C(C)c1cc[nH]n1)=O C1(O)(C(C)NC(c2ccc(C(C)C)s2)=O)CCN(C(C2CC(C)CO2)=O)CC1 CCCCS(=O)(=O)NCC(=O)NC1COCC1NC(C12CC(CN1C1CC1)C2)=O C1(NC(c2c(CC)nn[nH]2)=O)CN(c2nnc(C)s2)CC12CCOCC2 c1(C(=O)NCC(CC)NC(c2c(C)ccc(C)c2N)=O)cc(F)c(C)cc1F C(=O)(C(=O)C(C)CC)N1C(C)(C(=O)NCCSCC#C)C=CC1 c1(C(N2C(C)CC(NC(CCCOCCC)=O)C2)=O)nccc2ccccc12 c1(C(=O)NC2C(CNC(c3cc(C)sc3C)=O)CC2)c(O)nc(=O)n2c1CCC2 N1(C(CCc2c(C)noc2C)=O)CCC(NC(=O)CCCC2CCC2)C(C)(C)C1 C1(C(N2CC3CC3(CNC(=O)CC34CCCC3C4)C2)=O)(OCC)CCCCC1 N1(C(C2CC(=O)C2)=O)CCOC(CNC(C2(c3cccs3)CCCCC2)=O)C1 C1(C(N2CC(CC)(CO)C2)=O)CN(C(=O)CCC(=O)NC)CC1C N1(C(c2cnc(C)n2C)C(=O)NC2COC2)CC(C)(C)OC2COCC12 n1(CC)cc(Br)c(C(=O)NCCC2CCN(C(C3CC3(C)CC)=O)CC2)n1 CCS(=O)(=O)CCC(N)C(=O)NCc1ccccc1OCc1cccnc1 Cc1c2ccc(NC(C3(Cc4ccncc4Br)CC3)=O)cc2nn1C N1(C(=O)CNC(=O)C(F)(F)F)CCN(C(=O)CC2(O)CCC2)C2CCCCC12 O=C1CN(C(=O)C(=O)N(Cc2ccc(Br)cc2)Cc2cccnc2)CCN1 C1(C(=O)NCc2nc(C)c(C)[nH]2)C2CCC(C2)C1NC(=O)C1=CCCC1C C1(NC(C(C)NC(N)=O)=O)COC2C(NC(c3cnn4ccn(C)c34)=O)COC12 Cc1c(C(=O)NCC2CN(C(c3cc(C)n(C(C)(C)C)n3)=O)C2)cccc1O c1(C(N(CC(=O)O)Cc2cn(CC(C)C)nn2)=O)cc(-c2ccncc2)nnc1O C(N=c1[nH]ccnc1F)C1C(C)CN(C(=O)C=CCO)C1 c1(CC=C(C)C)ccc(C(N2CC(O)CC2CNC(C2(C)COC(=O)C2)=O)=O)nc1 c1(C(=O)NC(CCNC(C2ON=C(C)C2)=O)C)coc2c(Cl)cccc12 c1(C(=O)NC2CN(C(c3c(CC)nccc3)=O)CC2C)ccn(C)c(=O)c1 c1(C(=O)NC2CC(C)(NC(Cc3scc(C)c3)=O)C2)c(N)cc(Cl)nc1Cl CCC(CNC(=O)C(CC(C)C)ONC(C1CCCSC1C)=O)(CC)CO C1(NC(CCC(C)SC)=O)CN(c2nc3ccccc3s2)CCC12CCOCC2 c1(COC)nn(C)cc1C(=O)N(CCCN(C(=O)CCC1(C)CC1(F)F)C)C c1(CC(=O)NC(C(C)C)CNC(=O)CCOC2CC2)cccc(N2CCCC2)c1 N#Cc1cc(NC(c2cncc(-c3ccsc3C#N)n2)=O)cnc1Cl C1(NC(=O)CC2C=CCCC2)CC=C(C(=O)N2CC(CO)(CO)C2)C1 CN1CC(CNC(c2nc(-c3ccccc3)n(-c3ccccc3)n2)=O)CC1=O c1(CN(C2CCCCC2)C(C(C)OC(=O)CC2(C)CCCC2)=O)ccccc1Cl N1(C(COCCC)=O)CCC(OCCNC(=O)CC(C)c2ccco2)C1 Cc1cc(F)cc(C(=O)NCC2CCN(C(C3(C)CC3C)=O)CC2O)c1N C1(C(=O)NC2CC(C)(C)C2)CCN(C(c2cnco2)=O)CCO1 C(=O)(C(C)(C)S(C)(=O)=O)N(CCOCCCN(C(C)=O)C)C C1(C(c2nnnn2C(C)(C)C)NCC2CC(C)C2)CCC2CC1C2(C)C N1(C(=O)NCc2c(C)sc(Br)n2)CCc2ccc(Br)c(Cl)c2C1 c1(OCC)cc(C(=O)OCC2CC2n2cc(Br)cn2)ccc1OC(C)C C1(NC(=O)CCCNC(c2ccccn2)=O)CCCN(C(C2CC2F)=O)C1 C=C1CC2CCC(C1)N2C(=O)CCC(CC)NC(c1csc(C)c1)=O C(=O)(C(C(C)C)c1cccnc1)NCC1CC(NC(CSCCCC)=O)C1 c1(CC(C(=O)NCCCC(C)NC(CCSC)=O)C)cccc(F)c1 CC1C(NC(=O)CC2CCCCC2O)CCCN1c1cncc(C#N)n1 CCC(C)C(=O)C(=O)NC(CC1CCCO1)C(=O)NCCc1n[nH]c(C)n1 C(CC(C(C)C)NC(=O)C=C1CCC(C)CC1)NC(C(C1(O)CCCCC1)CC)=O N1(C(c2ccc(OC)c(F)c2)=O)C2CCN(C(C3CCCS3(=O)=O)=O)CC1CC2 C1(NC(C2CCCOCC2)C)CCCc2ccc(Br)cc2C1 c1(C(N2C(C)CC(CNC(=O)C(F)=CC3CC3)C2)=O)cnc2cnc(Cl)cc2c1 C1(C(N2CCC(O)(CO)C2)=O)CCN(C(c2ccsc2Cl)=O)CCO1 CC1=NOC(C(=O)NCC(C)(F)CNC(=O)C(n2nccc2C)C)C1 N1(C(Cc2ccc(C)c(F)c2)=O)CCC2(CCCN2C(=O)C(C)C2CCCC2)C1 N1(C(Cc2c(C)cco2)=O)CCn2ncc(S(C)(=O)=NC(=O)CC(C)O)c2C1 c1(C(N2C(C(N3C(C)C(O)CCC3)=O)CC3CC32)=O)cnc2ccc(F)cn12 C1(NC(C(C#C)(C)C)=O)CC2(CCC(CNC(C3CCN(C)C3=O)=O)OC2)C1 CCCCCC(O)CC(=O)NCC(CC)NC(c1cncc(C(=O)OC)c1C)=O N1(CC)CCCC(C(=O)NCCCCCCNC(=O)CC2CCC(=O)O2)C1 N1(C(C2C(C)=CCS2)=O)CCCCCCC1C(N1CC(n2cnnn2)C1)=O c1(OC)ccnc(C(=O)NC2CC(O)(CNC(c3n[nH]c4c3CCC4)=O)C2)c1O c1(OC)ccc(C(=O)NCc2ccc(CN(n3cccc3)C(C)=O)cc2)cc1 Nc1c(C(=O)NC2CCCC(NC(c3csc(Br)n3)=O)C2)cccc1Cl n1(CC)cnc(N=c2nc(C3CC3)o[nH]2)c1.CC=CC c1(CCC(=O)NCC2C(NC(C=C(C)Cl)=O)COC2)nc(C)c(C)o1 C1(C)(CNC(C(C)NC(C)=O)=O)CCN(C(=O)COCCc2ccccc2O)C1 C1(NC(=O)C(F)CC2CCCCC2)CS(=O)(=O)CC1N=c1[nH]nc(C2CC2)s1 N1(C(CCc2n(CC)ccn2)=O)C2CCC1CC(NC(c1nc(C)sc1C)=O)C2 c1(C(=O)NC2C3CN(C(c4sc(CC)c(C)c4)=O)CC32)cn(C)c2ccccc12 CC#CCC(C(=O)N(C)CC1CCCCC1)NC(=O)CCc1cnco1 S(=O)(=O)(c1ccsc1C(N1CC(NC(C2CCCCO2)=O)C(O)C1)=O)N(C)C c1(OC)cccnc1C(=O)N(CCCNC(C1CC(CC)=NO1)=O)C1CC1 c1(C(=O)NCCN(C)C(C2CCCS2)=O)oc2ccccc2c1CS(C)(=O)=O C1(C#N)(C(N(C(c2ccccc2)CNC(C2CCS(=O)(=O)N2)=O)C)=O)CC=CC1 C1(CC=C)(Cc2cn(CCCCNC(=O)CC)nn2)CCN(C(=O)CCCC)C1 c1(C(N(C(C)CNC(=O)Cc2sccc2C)CC)=O)cncc(C)n1 c1(-c2nc(CSC)nn2C2CCOC2)cc(F)cc(Br)c1F C1(NC(CC2C(C)(C)CC2)=O)CC(F)CN(C(=O)CSc2ccccn2)C1 N1(C(C(N2CCCC(C)C2)=O)=O)CC2CC(O)C1C2CNC(=O)C(F)(F)C(F)F C=CC(CC)CC(=O)N1CCN(C(=O)CN2CSCC2=O)C(CCOC)C1 c1(C(CC)(O)C(=O)N(c2cnc(C#N)cn2)CC)cccc([N+](=O)[O-])c1 N1(c2cc(C)ncn2)CCCC12CCCN(C(=O)C1=CCCCO1)C2 C1(O)(CNCC2CC3C=CC2CC3)CCCN(C(=O)OC)C1 N1(C(C(CC#C)C)=O)CC=C(CNC(c2cc(C3CC3)ncn2)=O)CC1 c1(C(N(CC(CNC(CC2(C=C)CCC2)=O)O)C)=O)cc(C)c(Cl)cc1OC C1(C(=O)NCC2CCCN(CC(C)C)C2)C(c2ccccc2)C2CC1C(O)C2O C(C1=NOC2CN(C(=O)Cc3coc(C(F)F)n3)CC12)NC(CCSCCC)=O c1(OC(C)C)ccc(C(C)OC(N2CCC(C)(O)C2)=O)nc1 c1(C(C(=O)N(CCC(C)NC(=O)CC2(O)CCC2)C)(C)O)ccc(Cl)cc1 C(CCCOC)(C(=O)N1CCC(F)(CF)C1)NC(C=NOC)=O N1(C(C(F)=CCC)=O)CCC(C(=O)NCC23CCC(CC2)O3)C(C)(C)C1 CC1CC(CNC(=O)C(c2ccccc2)F)CN(C(c2cnc3n2CCC3)=O)C1 c1(C(=O)NCC(N(C(c2cc(OCC)n[nH]2)=O)C)C2CC2)nccnc1C C(=O)(C1=CCC2(COC2)OC1)N1CCN(C(C2C(=C)CC2)=O)CC1 S(=O)(=O)(C(F)(F)F)OCCOC(c1ccc(CO)cc1)=O.C1(O)CCC1OO c1(CC(=O)NCCC(C)NC(=O)CN(C)C(N)=O)ccc(C(F)(F)F)cc1 N1(C(CCCc2nc(C)sc2)=O)CCCC(CCNC(c2cnc(Cl)s2)=O)CC1 c1(CN(C)C(C2(O)CCOC2)=O)ccc(CNC(c2coc(Br)n2)=O)cc1 c1(C(=O)NC2C(C)(C)CN(C(C3CSC3)=O)C2)cc(S(=O)(=O)N(C)C)c[nH]1 N1(C(c2cc(C)nc(O)n2)=O)CCC2(CC1)CC2NC(=O)CN1CC(=O)NC1=O n1(CCC)nccc1C(N1CCCC1CCCNC(c1cnc(OC)s1)=O)=O N1(C(CC(C)(C)NC(C)=O)=O)CCOCC(C(N2CCC3CC23C)=O)C1 CN1CCN(C(=O)CC2CC(O)C2(C)C)C(C(N2CCC(c3nn[nH]n3)C2)=O)C1 Cc1cc(C(=O)NC2CCC(F)(CNC(C3(CF)CC3)=O)C2)ncc1F c1(OC)cc(C(=O)NC2=CC=C2Cl)c(-c2ccc(C(C)=O)s2)cn1 N1(C(c2cc(CO)[nH]n2)=O)CCCN(C(=O)C(c2ccc(Br)cc2)O)CC1 c1(C(=O)Nc2cccc(OCc3cccnc3)c2)cc2ccc(Br)cc2nn1 CC(C)CC(CNC(C1CC(C)CCO1)=O)C(=O)NCCCC1C=NNC1=O c1(C2(NC(=O)NCC3(NC(C(CC)C)=O)CCCC3)CC2)c(C)noc1C c1(C(=O)NCC23CC2CN(C(c2n[nH]cc2[N+](=O)[O-])=O)C3)cnc2ncccn12 c1(C(=O)NCC2(CCNC(C(C(C)O)N(C)C)=O)CC2)ncc(Cl)c(N)c1Cl CC1(O)CON(C(=O)C2(CNC(=O)CC3CCCC4CC34)CCCO2)C1 c1(-c2nc(C(=O)NC(c3ccncc3)CC)sc2)c(F)cc(F)cc1F CC(O)C(C)(C)CNC(=O)C(c1ccco1)NC(=O)Cn1cnnc1O N1(c2c(Br)cnc(OC)n2)C2CCC1CN(C(C1CC1(Cl)Cl)=O)CC2 c1(C(N2CCCC(CNC(c3cc[nH]n3)=O)C2)=O)cc2cccn2cn1 C1(C(=O)NCCNC(C(CC)=CC)=O)CCCN(C(C2CC(CC(F)F)C2)=O)C1 C(=O)(C1=CCCOCC1)NC1(CC=C)CCCN(C(C2CCCN(C)C2)=O)C1 C1(C(=O)NC2(C(=O)NC3CCC(CO)CC3)CC(O)C2)CC1C1CCOCC1 C1(C(=O)OC2CN(C(=O)OC(C)(C)C)CC(F)C2)Cc2cc(Br)ccc2O1 N1(C(c2c(CC)nns2)=O)CCC(C(=O)NC2CCCCCC2F)C12CC2 c1(C(=O)NC2CC3(C(NC(CC(CC)C)=O)C3)C2)ccn2cnnc2c1 c1(SC)cc(C)ccc1C(=O)N(C1CCN(C(=O)Cc2cn(C)nc2C)C1)C CC1COCCCN1C(=O)CCC1CCC(NC(=O)CC2C(C)(C)C2(C)C)C1 CC1(C)CC(C)(NC(=O)C(c2cccs2)NC(=O)CN2CCNC2=O)C(=O)O1 c1(CC)csc(CNC(=O)CNC(C2CCC(F)C2)=O)n1 C1(C(N2CCC(N(C(c3n[nH]c(C)c3Cl)=O)C)CC2)=O)CCC12CCCO2 C(=O)(C(CNC(=O)CC1CCCCN1C)CC(C)C)N(c1cn(CCC)nc1)C N1(C(CN=S(C)(C)=O)=O)C2CCC1CN(C(C1CC1C1CCCC1)=O)C2 C1(NC(c2ccc(OCC(C)C)cc2)=O)CC2CCC(C1)C2NC(=O)CN(C)C C1(C(=O)NC(CC)CNC(=O)Cc2ccn(C)n2)OCCOC1(C)C C#Cc1ccc(C(=O)NC2CC(C(=O)NCC34CCC(CO3)C4)C2(C)C)cc1C CCC(O)C(C)(C)C(=O)N(C)CCN(C)C(c1csc(Cl)c1)=O Cc1c(Br)ccc(C(=O)NC2C3CN(C(c4c(C)cc(Br)cc4C)=O)CC23)c1F C1(OC)CC(CNC(=O)CCc2ncc[nH]2)N(C(C2CC(C)CCO2)=O)C1 N1(C(C2CC(OC(C)(C)C)C2)=O)CCCC(CNC(=O)NC2CCOC(=O)N2)C1 c1(OC)cc(F)cc(C(=O)NCC2CC(NC(c3cncc(C)n3)=O)C2)c1N C1(NC(C2CC(C(N)=O)C2)=O)CCCCC1C(N1CCCC1)=O.C12CC1C(=O)NC2 C1(OC)CN(C(C2CCC=CCC2)=O)CC1NC(c1cnc(C)n1C(F)F)=O C1(C(=O)NCCN(C(=O)CCc2ncccn2)CC(C)O)CC(O)CN1C C12(C(=O)Nc3ccc(C)cn3)CCC(NCc3cnc4ncccn34)(CC1)CC2 N1(C(CC2CCN(C)C2)=O)CCC(CNC(=O)CN2CCCCC2)C(F)(F)CC1 N1(C(CCOC(C)C)=O)CCN(C(=O)CCC(C)(F)F)CC1c1cccc(F)c1 Cc1cccc(C(=O)NC(C)C(=O)NC2C3CN(C(C4(Br)CC4)=O)CC23)c1 N1(C(N(C)CC2CCN(CC)C2)=O)CC2CCCCC12 c1(CC(N2C3CC(NC(C=C(C)C(=O)O)=O)C(C3)C2)=O)c(F)cccc1F C(=O)(C(C)(C)C(F)(F)F)N1CCC(C(=O)NCC2CC(=O)N(C)C2=O)CC1 CCCCCC(O)CC(=O)N1CC(OC)C(NC(c2nccnc2CC)=O)C1 c1(C(N(C(CCNC(CC2CC(C(=O)OC)C2)=O)C)C)=O)ccc(Cl)c(Cl)c1 c1(C(=O)NCC(CNC(CCCOCC=C)=O)CO)nn(C)c(Br)c1C c1(C(CC(=O)NC(CC(C)NC(c2ccncn2)=O)C)C)ccc(Cl)cc1 C1(NC(=O)NCc2c(C)c(Br)cnc2)CC(F)(F)CCC1(C)C N1(C(c2c(C(C)C)cco2)=O)CCC2CC(NC(C34CC(CO3)C4)=O)CCC2C1 c1(CC(=O)NC2CCCN(C(c3oc(C)c(CO)c3)=O)C2)cnn2ccccc12 C#CCC(CC(=O)OC)NC(=O)CCCN(C)C(C1(C(N)=O)CCC1)=O C(=O)(C1=CCCN(C(C23CCC(C2)C3)=O)C1)NCC(CC(C)O)C CS(=O)(=O)c1ccnc(NC2CCCN(Cc3cc4cc(Cl)ccc4[nH]3)C2)n1 c1(C(=O)NC2CCN(c3ncccn3)CC2)cccc2cnsc12 c1(C2(C(=O)NCCCc3cc(C(=O)O)no3)CCC2)c(F)cccc1F C(N=c1cc(C)nc(C(C)(C)C)[nH]1)C1CN(C(C(CCC)(C)C)=O)CC1(C)C C(=O)(C1CCc2cccnc21)N1CCC(C(C)(C)NC(CCC(N)=O)=O)C1 C1(CNC(CCNS(CC)(=O)=O)=O)COC(C)(C)CN1C(=O)Cc1cncn1C N1(C(CC2CCN(C)C2=O)=O)CCCC(C)(CNC(=O)COCC2CCCC2)C1 CCCCCCCCC(F)C(=O)NCCC(C)NC(=O)Cn1ccc(C(F)F)n1 C(=O)(C1=CCCCCC1)N(CC(=O)NCC1(C)CCC(=O)N1)CC1CC1 Cn1cc(C(N2CCC(O)(CNC(c3ccccc3)=O)C2)=O)c(Br)n1 c1(C(N2CCN(C(c3ncc(C)nc3)=O)CC2)=O)cc(C)c(C)c(F)c1 Cn1c(=O)c(CNC(C2C3CNC2C3)=O)cc2ccccc12 C1(CC)CCCCC1OCC(=O)NCC1(O)CN(C(C2(c3cc[nH]n3)CCC2)=O)C1 C(=O)(C1CCCn2cncc21)N1C(CNC(c2oc(C)c(Br)c2)=O)CC1 c1(N(C)C)ccc(C(=O)NC2CN(C(=O)CC3COCCO3)CC2O)c(F)c1 CCCN=C(NCc1cnn(CC(F)(F)F)c1)NC1CCC(OC(F)(F)F)CC1 N1(C(CCSCC)=O)CCCC(CN(C(C2C3(CC3)C23CC3)=O)CC)C1 c1(C(CO)NC(=O)NCC2CCC2O)ccccc1C(F)(F)F c1(C(N(C(C)C)Cc2cn(-c3ccsc3C(=O)O)nn2)=O)cnc2c(c1)ncn2C c1(C(C(=O)NCCCCCC)N(C(C)(C)C)C)ccc(Cl)c(F)c1 c1(C(N(C2CCC(O)CC2)C)=O)ccc(S(C)(=O)=O)[nH]1 C12(C(=O)NCCOCCCNC(=O)CC3CC(CF)C3)CCCCC1C2 Cc1cc(C(N2CCC(C(C)NC(c3cncc(N(C)C)c3)=O)CC2)=O)cnn1 C1(C(=O)NCC(C)CN(C(=O)CC2(O)CCCCC2)C)CC=CC(O)C1 CCC(C)CC(C(=O)OC)NC(=O)NCCOC(C)C C1(C(=O)NCC2(C(=O)NC(C3CCCCC3)C)CC=CC2)CCCC(=O)C1 C(CC(C)C(=O)OC)OC.n1(C2(C(=O)OC)CC2)cc(C(=O)NC2C3CCC32)nn1 C1(NC(C(C(C)C)C)=O)CN(C(=O)CNC(C2CCCCC2)=O)CC2CC12 C1(CNC(C(N2CCOCC2)C)=O)CC2CCC(C1)N2C(c1nnn(C)c1N)=O C(CC(C)(C)C(=O)NCCCCCCNC(c1cnc(C)cn1)=O)SC C#Cc1cc(C(N2CCCCC2CN(C(=O)C2=C(Cl)CC2)CC)=O)ccc1C C1(C(C)NC(c2ccc(C(F)(F)F)s2)=O)CCCCN1C(=O)COCCCF Cc1cnccc1CCNC(=O)CCCN(C)C(C1CCN(C)C1C)=O CC1OC2CCC1(NC(=O)C(C)CNC(=O)C(C)(C)CO)C2 C1(C(F)(F)F)(C(=O)OC)CCC(C(=O)Nc2cccc(C3(C)CCO3)c2)CC1 N1(CC(C)Nc2ccco2)CCN(c2ncco2)CC1 Cc1ncc2cc(C(=O)NC3CCN(C(c4ncncc4Cl)=O)C3)c(O)nc2n1 c1(C(N2CCC(C(C)NC(C3(C=C)CCC3)=O)C2)=O)cnc2c(c1)C(=O)CCC2 Cc1ncc(C(N2CCC(CN(C(=O)CC3CC=CCC3)C)C2)=O)cc1N Cc1cc(CC(=O)NCCC2CCCN2C(c2nccs2)=O)cc(F)c1 C(C)(CO)(C(=O)NC1(CC(=O)NCCC2(O)CCOC2)CC1)OC C(=O)(CCP(C)(C)=O)N1CC(NC(c2n(C)ncc2C2CC2)=O)(CO)C1 c1(OCC)cc(=NC(=O)c2csc(=NCc3ccnc(Cl)c3Br)[nH]2)[nH]o1 N1(C(CN(C2CCCC2)C)=O)CCC(NC(=O)C(C)(C)C2CCOC2)C(O)C1 Cc1coc(C(C)C)c1C(=O)NCC(C1CC1)NC(=O)Cc1csc(=N)[nH]1 N1(C(COCCOCC)=O)CCCC(C)C1CNC(C1CCOC(C)(C)C1)=O c1(CC)ccc(C(N2CCCC(CCNC(=O)C(C)OC(C)C)CC2)=O)cc1Cl N1(C(C(C)(C2CC2)OC)=O)CCC(NC(c2cc(C(N)=O)[nH]n2)=O)CC1 CN1CCOC(C(N2CCOCC(NC(=O)CSc3ccccc3)C2)=O)C1=O N1(C(c2c(NC)cncc2)=O)CC(CC(=O)NC2(CO)CCSC2)C2(CC2)C1 CCC1=C(C(=O)NC2CCCN(C(=O)C(C)CC(C)(C)C)CCC2)CCCO1 N1(C(C=C(C)C(C)(C)C)=O)CC(NC(c2c(C)oc(C)c2C)=O)CC12CCCC2 N1(C(CN(CCC)C)=O)CCCC(C2CCCN(C(=O)C=Cc3nccs3)C2)C1 C1(NC(CSCC)=O)CC(CNC(C2(C)CC2Br)=O)C1 C1(C(N(CCN=[N+]=[N-])CC)=O)CN(C)CCN1C(c1ncncc1N)=O N1(C(C(C2CC2)OC)=O)CCC2(CCCN2C(C2CCCC(C)CC2)=O)C1 c1(C(N2CC(NC(=O)CSc3nncs3)C2)=O)cc2ccccc2nc1C(F)F c1(OC)ccc(C(N2CC3CC2CC3NC(c2cnn[nH]2)=O)=O)c(OCC(F)F)c1 c1(C(N2CC(F)(CNC(CCNC(N)=O)=O)C2)=O)ccc(Cl)c(Br)c1F C#CCC(C)(C(=O)N1CCC(C#C)C1)NC(=O)C(C)N(C)C(C)=O N1(C(C2(C(C)(F)F)CC2)=O)CC2CCC(C1)C2CNC(=O)CSC1CCCCO1 C1(C(N2CC(C)C(N(C(=O)CC3(C)CCOC3)C)CC2)=O)CCCN2CCCC12 Cc1nn(C)c(Cl)c1C(=O)NC1CCCN(C(C2CCS(=O)(=O)CC2)=O)C1 N1(C(C(C)CC2CC2)=O)C2CCCC1CC(NC(=O)CSC(F)(F)F)C2 Cc1cc(C(=O)NCCN(C(c2cc(Br)n[nH]2)=O)C(C)C)nc(C(F)F)n1 c1(NC(C(=O)Nc2cnn(CC(=O)OC)c2C)=O)c(Cl)cccc1Br C1(CC(=O)NCCN(C(C(CCCC)C(C)C)=O)C)CCc2ccccc2C1=O C1(C(N2CCN(C(C#C)C)CC2)=O)CCCN1NC(=O)C(O)C=C CC(C)C(CC(=O)NCCC12CCCC1C2)NC(=O)CCOC1CCCC1 CCC(C)C(C)C(=O)N1CCCC(CN(C)C(c2nnc(CSC3CC3)o2)=O)C1 c1(OC)ccc(C(N2CCC(CNC(C3(CO)CCOC3)=O)C2)=O)nc1 c1(C(=O)NCC(CNC(C2CC23CC3)=O)C(F)(F)F)c[nH]c2cc(F)c(F)cc12 C1(NC(c2c(COC)cco2)=O)CCCN(C(c2cn(C)nc2C(C)C)=O)C1 N1(C(C(C)(O)C2CCC2)=O)CC2CCC2(CNC(=O)C(c2cccc(F)c2)F)C1 c1(SCC(=O)N(C)CCN(C)C(C2(C)CC2(F)Cl)=O)ccc([N+](=O)[O-])cc1 c1(C(c2nnnn2C2CC(F)(F)C2)NCCC(C)CO)ccccc1[N+](=O)[O-] N1(C(CC(C)F)=O)CC2CC2(C(=O)NC2CN(c3ncco3)C2)C1 c1(C(N2CC(C)(CCC(=O)NCc3ccc(Cl)cc3)C2)=O)cnc(O)c(F)c1 N1(C(c2c(C)nco2)=O)C(CNC(=O)CC23COCC(C2)C3)CC2CCCC12 C=Cn1nccc1C(N1CCC(NC(=O)CC(=O)N(C)C)C1C(C)(C)C)=O c1(OC)cc(CN(C(CC2CC2)C(=O)NC2(CC3CC3)CC2)C)ncn1 C1(C(=O)NC2(C(=O)NC3CN(C(C)=O)C3)CC2(C)C)CCCC(=O)N1 Cc1cnc(NCC2(C)CC2Br)c(S(=O)(=O)NC2CC=CC2)c1 N1(C(COCCOC)=O)CC(O)(C2CCN(C(=O)CC3=CCOCC3)CC2)C1 C(CN=C(NCC1CCCNC(=O)C1)N(C)Cc1ccc(Cl)s1)OCCOC Cc1nc(C(=O)NC(CC(=O)NCC2(CO)CC2(C)C)C(F)(F)F)ccc1C#N c1(-c2nc(CN(C(=O)CN3CC(N)CC(O)C3)C)on2)cc2scc(Cl)c2[nH]1 N1(C(CCOCCC)=O)CC2CC3CC2C1C3NC(c1ccc(F)cc1Cl)=O CC(C)C(O)C(C)C(=O)N1CC(C)(OCC(=O)NC2(C3CCCOC3)CC2)C1 C1(CNC(c2ccc(SC)o2)=O)CC(O)CN1C(=O)C(C(C)C)NC(N)=O N1(C(c2ccc(C(C)C)s2)=O)CCN(C(C2(C3CCOCC3)CC2)=O)CCC1C C1(N(C(=O)CCc2ccccc2)CCC)CCN(Cc2ccc(Cl)cn2)CC1 N1(CCCNC(=NCC)NC(c2ccnc(C)n2)C)CCc2ccccc2C1 N1(C(C2C(C)C2)=O)CCCC2(CCCN2C(c2cncc3c2CCCC3)=O)C1 c1(C(=O)OCC)nc(CNCC(c2cnccn2)C)sc1N Cc1nn(CC(F)(F)F)c(C)c1CC(=O)NC(c1cnc(Cl)cc1)(C)C C1(CNC(c2c(C)ncs2)=O)CN(C(=O)CCc2nnc(C)n2C)CC12CC2 C1(C)(CC)CN(C(=O)CC2CCC(NC(c3cc(Cl)cs3)=O)CC2)CCO1 c1(CCC)c(C(=O)NC2(C)CN(C(=O)C(C)Oc3ccc(F)nc3)C2)cnn1C C1(NC(=O)C(c2ccc(C(F)(F)F)cc2)O)CCCCNC1=O C12(NC(C3(C)C(C)(C)C3(C)C)=O)CCCN(c3ccccc3[N+](=O)[O-])CC1C2 C(CC(CC)C(=O)NCCCOCCC(=O)N(C(C(N)=O)C1CC1)C)=CC C1(C(N(CCCC#C)C)=O)C2CCC(C2)N1C(=O)C=CC1CCCC1 C(=O)(C(CCC1CC1)NC(=O)C(C(C)C)OC)NC(CC=C)CC CCC(CC(F)(F)F)C(=O)NCC(C)CN(C(=O)CS(=O)(=O)CC)C C(=O)(C(CCCC)C(C)C)NC1(CC=C)CCN(C(c2nc(C)ncc2Cl)=O)C1 N1(C(CCC=CC(C)C)=O)CCC(OCCNC(C2CC2C)=O)CC1 Cc1nc(-c2ccc(Cl)s2)sc1C(=O)N(C1CCN(C(=O)CCC(N)=O)C1)C C(=O)(C1=Cc2ccc(Cl)cc2OC1)N1CCC(CC=C)(NC(c2cnco2)=O)C1 c1(CC)nc2ccccn2c1C(N1CC2(CC(NC(=O)C(C#N)C3CC3)C2)C1)=O CC(F)CC(=O)N1CC(N(C(=O)C(C)C2CN(C(=O)OC(C)(C)C)C2)C)C1 Cc1cccc(C=CC(=O)NC(C)CCCC(=O)NC(C)CC(F)(F)F)c1 c1(CO)cc(ONC(C2(CC#C)CCN(C(=O)C(C)(C)C#CC)C2)=O)ccc1F C(C(=O)NOCC(F)F)=C(C)CN(C(=O)C(C1CCOC1)N(C)C)C Cc1cc(Cl)cc(C)c1C(=O)NCCC1COCCN1C(=O)CCS(N)(=O)=O c1(OC)ccc(F)c(Br)c1C(=O)NC1CC(O)CN(C(=O)C(F)=C(C)C)C1 C(CCCCCNC(=O)C(F)=CC1CC1)N(C)C(C1CCSC1)=O C1(NC(N2CCN(C(N3CCCC3)=O)CC2)=O)CCCC12CCC2 C=CCC(F)(F)C(=O)NCC(O)CN(C(=O)CCOCC1CCCO1)C C(CC(C(=O)N(C1CCCCC1)C)NC(c1coc(C2CC2)n1)=O)=CC c1(C(=O)NC2(CNC(c3ncc(C)cc3C)=O)CC2)cc(C)c2[nH]nnc2c1 C1(C(N(C2CCCN(C(c3ccc(F)cc3)=O)CC2)C)=O)CN2CCCC2CO1 c1(SC)ccc(O)c(C(N2CCC(CNC(=O)Cc3nccs3)C(C)C2)=O)c1 C1(NC(C(CC)N(C)C)=O)CN(C(=O)CCN2CCC(O)CC2)C2(CCCC2)C1 c1(C(N(CC(C)NC(=O)Cn2cnnc2)CC)=O)ccc(CO)cn1 C1(CC(=O)N(C2CN(C(CNC(c3ccc(C)s3)=O)=O)C2)C)CCCCCC1 c1(C(CNC(C#C)CO)O)ccc(Br)cc1 c1(CC(=O)NCC2CCCN2C(C2CCCCC(=O)N2)=O)cccc2[nH]ncc12 CN1CCC(CC(=O)NC2(C(=O)NCC3(C)CC4CC4C3)CCCC2)C1=O N1(C(C(C#C)(C)C)=O)CCC(NC(C2CC(O)(C(F)(F)F)C2)=O)C2(CCC2)C1 C(=O)(CC(C)C(=O)N1CC(C)(NC(C2COC(C)(C)CO2)=O)C1)OC N1(C(C(CC)NC(C)=O)=O)CCN(c2ncncc2C#N)C2(CC2)C1 C1(n2cc(-c3cc(CC)ns3)nn2)CCN(C(=O)CCCCCN(C)C)CC1C c1(OC)ccc(C=CC(=O)NC(C)CN(C)C(C2CCC(CO)CC2)=O)cc1F c1(NC(C=CC(C)NC(CCC(C)(C)OC)=O)=O)cccn2ccnc12 CCC(CC)C(F)C(=O)NCC1CN(C(=O)CC2CCOCC2)CC12CC2 c1(C(N2CCN(C(CC=C=C)=O)C(C(C)C)C2)=O)c(OC)ccc(SC)c1OC c1(C(N2CCCC(N(C(CCSC)=O)C)C2)=O)cccc(C)c1C#N C1(CCN(C(C(COC)O)=O)C)CCCCN1C(=O)CC(C)O C(=O)(C1=CCC(C)CC1)N(C1CCCN(C(=O)C(C)(C)n2ccnn2)C1)CC C1(C(=O)NCC(=O)NCCC)CCCC1CNC(c1csnc1C)=O C1(NC(Cc2ncc(C)s2)=O)CN(C(c2cccc(C3(C)CC3)c2)=O)CC1C C#Cc1ccc(C(=O)NC2CCCC2CNC(c2ccoc2CC)=O)c(F)c1 C(=O)(C1=C(C2CC2C)N(CC2CC2)C(=S)NC1c1cnsc1)OCC c1(NCCN(C(C2CC(C)OC2)=O)C)c([N+](=O)[O-])c(C(F)(F)F)nn1C N1(C(C(C2CCCOC2)NC)=O)CCN(c2ncc(C(=O)OC)s2)CC1 C1(C)(CNC(C(c2cnn(C)c2)C)=O)CCN(C(=O)CCC(C)(C)C)CC1 c1(C(=O)NCC(CC=C)NC(c2cn(CC(=O)NC)nn2)=O)cccc(CO)n1 c1(C(N2C(C)(C(=O)Nc3ccc(C#N)cn3)CC2)=O)cccc2oc(S)nc12 Cc1ccc(CC)c(C)c1.C1(NCC(=O)N)CCN(c2ncnc(Cl)c2F)CC1C c1(C(C(=O)NC(C2CCOC2)CNC(CN(C)CC)=O)(F)F)cc(F)ccc1F C1(SCCN2CC(=O)N(CCC=C)C2=O)CC(SC)C12CCCC2 C(C1CCCN1C(c1ccsc1)=O)=CC(=O)NCc1cnn(CCF)c1 c1(C(=O)NC2C(NC(CCc3onc(C)n3)=O)CCC2)ncc(Cl)c(N)c1Cl Cn1cc(CN2CC(F)(C(N3CCC(CO)C3)=O)C2)cn1 CC1CC(O)CCN(C(C23CC(C)(CN2C(c2ccsc2)=O)C3)=O)C1 c1cc(C2CCC2)ccc1N(c1cnn(C2CC3(CCC3)C2)c1)N1CCCC1 Cc1nc(C2CC2)oc1C(=O)NCCN(C(=O)CC1COCC(C)O1)C c1(CN2CCC(NCc3c(OC)cccc3)C2)c(F)cccc1Br c1(NC)ccc(C(=O)NCC2CCCCN2C(c2ccc(=O)n(C)c2)=O)cc1F CC1CN(C(c2csc(CNC(C3CCCCO3)=O)c2)=O)CCC1(F)F c1(C(=O)NCC2CC(NC(CN3CCC(C)CC3)=O)C2)cccc2c1OCC2C C1(C(=O)NC)CCN(C(=O)C(C2CCC2)NC(=O)C(C2CCC2)OC)CC1 CN=c1[nH]c(=NCC(C)c2cccc(Cl)c2)[nH]c(=NCC(C)(C)CO)[nH]1 C1(NC(C2CC3CCC(C2)O3)=O)C2CCC(C2)C1C(=O)NC1(CO)CC=CC1 N=c1nc(CCC(=O)NC2CC2NC(C2CCCN2C(c2cccs2)=O)=O)[nH][nH]1 C(=O)(CC(C)(C)Cc1ccccc1)NC(CCCNC(c1c(C)csc1C)=O)(C)C c1(NCc2nc(CC)sc2)ncnc(N2CCSC(C)(C)C2)c1C c1(C(=O)NC(C)C(C)NC(C2CCN(C)C2=O)=O)cc2c(C(F)F)nn(C)c2s1 C1(CNC(=O)Cn2ncnn2)CC2(CCOCC2)CN1C(c1cc(Cl)on1)=O C1(F)(C(N2CC(CNC(=O)CNC(=O)NCc3ccsc3)C2)=O)CCCC1 c1(C(=O)NCCC2(O)CCN(C(C(C(C)C)(C)O)=O)C2)cc([N+](=O)[O-])ccc1Cl Cc1cc(C(=O)NC23CC(NC(c4cc(=O)c(Br)c[nH]4)=O)(C2)C3)ccc1F C1(CNC(C2CC=C(C)CC2)=O)CN(C(c2cccc(N)c2C)=O)C(C)(C)C1 c1(NC(CC2(NCc3cc(C)c(Cl)nc3)CCC2)=O)cccc2cncc(Br)c12 N1(C(CC(=O)OC)=O)CCC2C1CCCN2C(=O)CC(c1ccc(OC)cc1)C CC(F)(F)C(C)(C)CC(=O)NC1CC(CNC(=O)Cc2n[nH]cc2Br)C1 N1(C(c2ccc(C)cc2C)=O)CC(NC(=O)CCN2CCCC2)CC(C)(C)C1 c1(CC(=O)NC2CC(CNC(C3(C)CCC(=O)N3)=O)CC2O)cc(F)cc(Cl)c1 CN=c1[nH]nc(CC(=O)N(C(C)CCNC(=O)C(C)(C)c2ccn(C)n2)C)s1 N1(C(c2cc(C(C)=O)[nH]n2)=O)CCCC(CCCCNC(c2ccoc2C)=O)C1 C1(C(N2CCC(CN=c3[nH]nc(C)o3)C2)=O)CC2(CCC(C(N)=O)CC2)C1 CCCC(CCC)C(=O)NC(C)(CSC)C(=O)NC(C(C)C)C1CC1 C1(C(=O)NC2CC3(CCC3)C2)(NC(c2cocn2)=O)CCOCC1 C1(NC(C(Cc2ccccc2)OC)=O)CNc2c(c(C)nn2C)C1.C1CC(=O)N1 c1(C(N2CC(NC(c3nnn(CC)c3C)=O)C(F)CC2)=O)cncc([N+](=O)[O-])c1 c1(C(N2CC(C)(CNC(CCOCC#C)=O)C2)=O)ccc2cccc(F)c2n1 N1(C(C(CC)OCC)=O)CCC(C)(CC(N2CCC(CC3CC3)C2)=O)C1 C1(NC(C2CC(F)(F)CS2)=O)C2CC1N(C(=O)CCc1ccncn1)C2 N1(C(=O)Cc2ccccc2Cl)CC2CCN(c3ncc4[nH]ccc4n3)C2C1 c1(C(=O)NC(c2ccccc2)CNC(C2(OC)CC2)=O)cc2cc(F)ccc2o1 C(C(CC(F)(F)F)NC(C1C2(CC2)C12CC2)=O)NC(c1c(C)nc(O)[nH]1)=O N1(C(c2c(COC)nn[nH]2)=O)CCC(C)C1C(=O)NOC(C)C(O)C(F)F CC1(NC(=O)C(Cc2cc[nH]n2)NC(c2n[nH]cc2Cl)=O)CCCOC1 C(=O)(CCCNC(=O)C(C)CNC(C1C=CCS1)=O)OC C1(N2CCN(Cc3c(-c4nccc(SC)c4)onc3C)CC2)CC(C)(C)OC1=O C=CCCC(C)N=c1nc(N2CCCC(N3CCCC3)C2)c2c([nH]1)CCCCC2 c1(C(N2C(C)(C)C(CNC(=O)CNC=O)CC2)=O)snc2ccc(Br)cc12 C(=O)(C(C(C)(C)C)N1CCNC1=O)NC(C)CCNC(c1cnn(CC2CC2)c1)=O C(C)(CCCNC(=O)C(C)(C)NC(=O)NC1CC1)NC(C1C(=C)C1)=O N1(C(CC(C=C)C)=O)CC2CCN(C(c3c4c(nn3C)CCSC4)=O)CC(C2)C1 C1(NC(CC2(C=C)CC2)=O)CCN(C(c2c(C)ccc3n[nH]cc23)=O)CC(C)(C)C1 C=CCC(CNC(=O)CN(C)C(C1CCC(C)(O)CC1)=O)CC(C)C c1(C(=O)NC)cccc(C(N2CCCC2C(C)NC(=O)CCC2(C)CC2)=O)n1 C1(C(N(CCCNC(c2c(OC)cccc2)=O)CCO)=O)CN(C)CCN1C C(c1ccccc1)=CCNC(C1C(C)CN1C(=O)CC1CCCCO1)=O c1(NC(C2CC(NC(c3nc4ccccn4n3)=O)C2)=O)nccc2cccnc12 CCC(C)(C)CC(=O)NCC1CC(NC(=O)C(C(C)C)N(C)C)C(O)C1 c1(C(=O)NC(C2N(C(CCC=C)=O)CCC2)(C)C)ccc(N2CCCC2=O)cc1 C12(NC(CC(C=C)C)=O)CCC(NC(C3CC(=O)CC(=O)C3)=O)(CC1)C2 Cc1ccc2c(C(=O)NC3CCN(C(=O)C(C)(O)C(C)(C)C)CC3C)c[nH]c2c1 n1(-c2ccn(C(C)C)n2)nc(-c2nccs2)nc1C(C1CCOCC1)F c1(C(N(CC)CC)=O)ccc(CNC(=O)CC2CC(C(=O)OC(C)(C)C)C2)cc1 [N-]=[N+]=Nc1ccc(NC(=O)CC(C(F)F)NC(C2CCC(F)(F)C2)=O)cc1 Cc1c(C(=O)NCC(C)(C)C(=O)NCC2CSC2)cccc1F c1(C(=O)NCC#CCNC(Cn2cc(C)c(C(F)(F)F)n2)=O)cncc(C)c1Cl C(=O)(CCCCC1CCCC1)N(C1CCCCC1)CCNC(C1CCN1CC)=O c1(C(=O)NC23CC(NC(C(C)N(C)C)=O)C(OC2)C3)c[nH]c2ncccc12 C1(NC(c2c(C(=O)OC)ccc(C)n2)=O)CCC2(CC1)CC2(F)F N1(C(c2c(CCC)occ2)=O)CC2(COC(CNC(=O)C(O)C(C)C)C2)C1 c1(C(N2CCC(CN(C(C3(C)CC(C)C3)=O)C)CC2)=O)[nH]nc2ncnc(O)c12 C1(C(=O)NN2CCC(C)C2)CCCNC1=O.C12CC(C1)CC(=O)N2 CC(C)C(O)C(F)(F)C(=O)NCCN(C(=O)C1=CCCC1C)C C(=O)(C(C)(C)S(=O)(=O)C1CC1)NCC(CNC(C(CC)N1CCCC1=O)=O)OC N1(C(C(C)NC(N)=O)=O)CC2CC(N(C(=O)CCCc3cnn[nH]3)C)C1C2 C1(CC(N2C(CN(C(=O)CCCC3CC3)C)CCC2)=O)CCc2sccc2C1=O c1(OC)ccc2c(c1)C(C(=O)N1CCN(C(C3(N(C)C)CCC3)=O)CC1)CCC2 CC1(CNC(C2(C3CCCO3)CCC2)=O)CCCN(C(c2nccnc2Cl)=O)C1 C1(C(N(OCC(=O)OC)C)=O)CCCCN(C(=O)COC2(O)CCCCC2)C1 N1(C(c2cc(C(C)=O)oc2C)=O)CC2COCCC2(NC(=O)C2=CCCCO2)C1 c1(CN2CC(C(N3C4CCC3CC(O)C4)=O)OCC2)cc(Br)cc([N+](=O)[O-])c1O C1(C#CC(=O)NC2(C)CN(C(=O)Cc3ccc(Br)s3)C2)(CC)COC1 N1(C(COCCCC#C)=O)CCC(C(=O)OCC(C2CC3C=CC2C3)=O)CC1 CCCCC(C)(F)C(=O)NCCC(F)Cn1cc(-c2ccc(N=[N+]=[N-])cn2)nn1 N1(C(CC)=O)CCN(C(=O)C(O)CC2CCOCC2)C(C2CCC2)C1 C12(n3cc(CC=C)nn3)CCC(C(N3CCC(C(O)C(F)(F)F)CC3)=O)(CC1)C2 c1(C(c2nnnn2C(C)C)NC(CSC)C)cnc(Br)s1 c1(C(=O)NCc2c(CNC(CN(C)CC)=O)nccc2)cnn2c1C(=O)NCC2 C1(SC)CN(C(c2ccn(CC(=O)OC(C)(C)C)n2)=O)CC1NC(=O)C=C(Cl)Cl C1(SC)CN(C(=O)C(C)(COC)OC(C)=O)CC1n1cc(C(C)(C)O)nn1 N1(CCc2c(CC)cccc2)CCC2(NC(c3sccc3C)=O)CCCC12 CCCCCC(C)CC(=O)NC1CC2CCC(C1)N2C(C12CC1COC2(C)C)=O c1(COC)nc(NC(COC)C2CC2)cc(=NCc2cccc(N)c2C)[nH]1 C1(O)(CNC(C(CC)OCC)=O)CCN(C(c2n[nH]c(C)c2F)=O)C1 C1(CNC(=O)Cc2cc[nH]c2)CC2(CC2)CN1C(C1CCSCC1)=O C1(CC)CC12CCN(C(=O)CSC)CC2.c12conc1C(=O)NC2c1cccs1 N1(C(c2nc(C)n(C)c2)=O)CCCC12CCCN(C(=O)Cn1cncn1)C2 C1(OC)CC(C(=O)Nc2ccc(Cl)cc2)N(C(=O)CCc2cncs2)C1 C1Cc2[nH]c(=NCC3CN(CC4CC4)C3)[nH]c(=NC3CC(=C4CC4)C3)c2C1 C1(C)(CC)CCCN(C(=O)CC(C(C)C)NC(c2cc(C3CC3)on2)=O)C1 c1(C(=O)NCCNC(c2cc(CC)oc2C)=O)ccc(-n2cnnn2)cc1Cl C1(C(N2C(C)CC(NC(C3C4CC5C(C4)C35)=O)CC2)=O)CC2CC1CC2(F)F C1(CNC(c2ccn(C)n2)=O)CCN(C(C2C(C#N)C2(C)C)=O)C12CCC2 C1(CNC(=O)C(F)n2ccnc2)CN(C(c2ccc(F)s2)=O)CCO1 C=C=CC(C)C(=O)NC(C)CN1CCN(C(=O)C(=Cc2ccncc2)C)CC1 C(C(=O)NNC(=O)Cc1ccccc1)NC(Cc1cccc(OC)c1)=O C(=O)(C(C)(C)C1=CCN(C(=O)CSC(F)(F)F)C1)N1CCN(CC)CC1C N1(C(C(C)c2ccsc2)=O)CC(C)N(C(=O)CCc2ccccc2)CC1C N1(C(C(C)SC(C)C)=O)CC(CC(N2CCNC(=O)C2CCO)=O)CC1(C)C CCCCC#CC(C)(C)NC(=O)CCCCNC(C1OCCC1C)=O C1(NC(COC(CC)C)=O)(CF)CCN(C(c2ccc(C(F)F)s2)=O)C1 C12(C(N3CC(NC(C4(C)CC(=C)C4)=O)C3)=O)CC(CO)(C1)OC2(C)C C(=O)(N=c1[nH][nH]c2ncccc12)C1C2CN(Cc3c(COC)nn(C)c3)C1C2 N1(C(C2CC3C(C)(C)C3C2)=O)CC2(CCC(NC(C3C4COCC34)=O)CC2)C1 CN1CCCC(F)(C(=O)N(CC(C)(C)CNC(C2(C)CCOCC2)=O)C)C1 c1(NC(=O)CCCN(C(=O)C2=C(C)CCCC2)CCC)ccc2c(c1)CCC2 c1(COC)ccc(-c2cn(CC3CCCCN3C(=O)C(C)C(F)F)nn2)cc1 Cn1cc(N)c(C(N2CC(F)(CNC(c3ccoc3Cl)=O)C2)=O)n1 C1(NC(c2nn(C)c(Cl)c2)=O)COC2(CCN(C(=O)C=Cc3cnccn3)C2)C1 C1(O)(CCNC(c2ccc(OC)nn2)=O)CCCN(C(c2cncc(O)c2)=O)C1 N1(C(c2cc(C)c(C)nn2)=O)CC2(C(=O)NC(C)Cc3cn[nH]c3)CC1CCO2 C1(CNC(C(CC)c2ccccc2)=O)CC(O)CN1C(=O)C(C)NS(=O)(=O)CC C=CC(COC)N=c1nc(N2Cc3cc(O)nnc3C2)c2cc(Cl)ccc2[nH]1 Cc1cccc(OCC(=O)NC2CCN(C(=O)CCN3CCCCC3)C2)c1 C1(NC(c2ccn(CCNC(=O)C(F)(F)C3CC3)c2)=O)CCCC2(C1)N=N2 C(C(=O)N=c1ccn(CC2CC2)[nH]1)C1N(C(CCCC(=C)C)=O)CC(O)C1 N1(C(C(C(C)C)CO)=O)C2CCCC1CN(C(C1(C(=O)NCC(F)(F)F)CC1)=O)C2 c1(C(N2CC(CC)N(c3cc(C#N)ncn3)CC2)=O)cc2[nH]ccc2cc1OC N1(C(C2C(C(=O)OC)C2)=O)CCSCC1CCNC(=O)CC1CCC2CC12 CCC(C(=O)NCCCOCCN(C)C(C1CCOC(C)(C)C1)=O)C(C)(C)CC N1(C(c2nc(OC)oc2)=O)CC2CC(NC(c3ncccc3C)=O)C1C2 c1(C(N2CC(OC)C(NC(=O)Cn3nnc(=O)[nH]3)C2)=O)nn(C)cc1S(N)(=O)=O c1(OC)sccc1C(=O)NC(C)C(C)NC(c1coc(C)c1)=O N1(C(C=C(C)C(C)C)=O)CCCC(CNC(=O)Cc2cnc(C)[nH]2)CC1 C1(CNC(C(=Cc2cccnc2)C)=O)C(C)CCCN1C(c1ccccn1)=O N1(C(C2CCC(=O)N2)=O)CCC(CNC(c2ccn3ccnc3c2)=O)C(F)(F)C1 N1(C(C=C(CC)C)=O)CC(OC)C(NC(c2cncc(CN(C)C)c2)=O)C1 c1(C(=O)NC2COCCN(C(c3cccc(Cl)c3)=O)C2)ccc2nnc(S)n2c1 c1(C(N(C2CC23CN(C(=O)OC(C)(C)C)C3)C)=O)cc([N+](=O)[O-])c(O)cc1N C1(C(N(C(C)C(=O)N(C)C)C)=O)(CNC(C2CCCC(CF)C2)=O)CCCCC1 CCCC(O)CC(=O)N1CC(F)(F)CC1CCNC(c1coc(C(C)OC)n1)=O Cc1cn2cc(NC(C3CC4(CC4)CN3Cc3ccc(Br)cc3C)=O)ccc2n1 C1(CNC(C(CC)OC)=O)CN(C(c2c(C)noc2C)=O)CC1O c1(CN2CC(CC)N(C(C3CCCN3C)=O)CC2)cccc2c1OCO2 C12(NC(c3nc(COC)sc3)=O)CCCC1N(C(=O)CCc1ccnn1C)CC2 c1(CN(CC(N2CCCN(CCC#C)CC2)=O)C)cnc2sc(C)c(C)n12 O=C(O)C(NNc1ccc(F)nn1)c1csc2cc(Cl)ccc12 C1(c2c(C)cc(Cl)nc2)NC(=S)N(CCOCCO)C2=C1C(=O)NC2c1ccccc1 Cn1c(=O)cc(-c2nc(Cc3cccc(F)c3)no2)c2ccccc12 N1(C(C(C)C(C)c2ccc(F)cc2)=O)CC(NC(C2(O)CCC2)=O)C(C2CC2)C1 c1(CNC(N2CCC(CCC(F)(F)CO)C2)=O)ccnc(Br)c1F C1(N(C(C(=O)NCCOCC)=O)C)CCc2nc(C)nc(C(F)(F)F)c2C1 c1(N(C)C)ccc(Nc2nnc(C(F)F)o2)c(C(F)(F)F)c1 c1(NC(N2CC(CC)N(C3CC3)CC2)=O)ccc(NC)c2ccncc12 C=CC(CC)CC(=O)N1CC2CC2(NC(=O)CCCc2cccc(Cl)n2)C1 C1(C(=O)NC(C=C)C)C2CCCC1CN(Cc1cccc(Cl)c1Br)C2 C1(C(C)O)CCC(NC(C2(N(C)C(c3c[nH]c(=N)o3)=O)CC2)=O)CC1 c1(SC)nccc(=NC2CCC3(C2)CN(C(c2ccc(Cl)c(O)c2)=O)C3)[nH]1 CC(C)CC(C)(C)C(=O)NCC12CC(NC(=O)CN3CCCC3=O)(C1)C(C)O2 C1(CNC(N(C)CC(CCC)OC)=NCC2CCC2)CC2(CCC(CO)CC2)C1 C(=O)(C(CCCC=C)NC(C1OCCC1C(C)C)=O)NC1(C#C)CCCCC1 N1(C(CCOCC#C)=O)CCN(C(c2ccc(C(F)C(F)(F)F)cc2)=O)CC1 c1(C(=O)NCC(C(C)(C)C)NC(c2cc(C)cc(O)n2)=O)cc(C)c(C)nc1O c1(C(CC(=O)N(C2CSC2)OC(=O)OC(C)(C)C)CC)ccn(C)c(=O)c1 C(=O)(C#CC1(C)CCCO1)N1CCN(C(CCC(C)(C)F)=O)CC1CO c1(C(c2nnnn2C2CCOC2)NCCC=C)ccc(C2CCC2)nc1 Cc1cc(NC(=O)C(C)NC(=O)C(N2CCNC2=O)C)cc(C)c1F c1(C(=O)NC(CCNC(C2CCCN(CC(C)C)C2)=O)C)cncc2ccsc12 c1(OC)ccc(CC(=O)NCCCCCNC(=O)C=Cc2cc[nH]n2)nc1 Cc1c(NC(=O)NCCC2(C)CC2(F)F)cccc1S(N)(=O)=O c1(CC(=O)NCC(C)NC(c2ncn(C)n2)=O)ccnc(F)c1F c1(NC(C)=O)cccc(C(=O)NC2CCCN(C(=O)Cc3cncn3C)C2)c1 CCCC(CCCNC(=O)C(=Cc1ccncc1)C)NC(=O)C(C(C)C)C1CC1 N1(C(C)=O)CCC(C)(C(=O)NCC(C2CC2)N(C(=O)CSc2nc[nH]n2)C)C1 C1(C(N2CCC(n3cc(CNC)nn3)CC2)=O)CCCCC(=O)N1 c1(C(N(CC(C)(C)CNC(C2(O)COC2)=O)CC)=O)ccc(C)c2ncccc12 C(C(C)(O)C(C)(C)C)NC(CCC1(C)CN(C(C2CC(C)(O)C2)=O)C1)=O C1(O)(CN(C(CN(C)C(N)=O)=O)C)CCN(C(=O)C(C2CCOCC2)O)CC1 C1(CC(=O)NCC2C(C(=O)NC(c3ncc(F)cn3)C)CCC2)CCCC2CC12 c1(C(N(C)CC2(NC(=O)CCc3ccco3)CC2)=O)cc2n(c1)CCOC2 CCCCC(=O)NC(Cc1cn[nH]c1)C(=O)NCCCC(=O)N(C)C C1(C(C)NC(Cc2c(C)scc2)=O)CCN(C(c2ccccc2C2CC2)=O)CC1 C1(O)(C(=O)NCCOCCN(C(c2ccn(COC)n2)=O)C)CCOCC1 C(=O)(CN=Cc1ccco1)N1CCC(O)(C(=O)NCc2ncn(C)c2)CC1 N1C(=NCCCN2CCOCC2)NCC1.Cc1cccc(C)c1Sc1nccs1 c1(C(N2CCN(C(C3(C)CCCN3)=O)CC2C(F)(F)F)=O)cc(Cl)cc(F)c1Cl N1(C(C=CCC)=O)CC(NC(=O)C(C)OCc2ccncc2)CC2(CC2)C1 CCCN=C(NCC1(S(C)(=O)=O)CCC1)NC1CCN(c2cccc(Cl)c2)C1 CCCCS(=O)(=O)CC(=O)N1CC2CC1CN(C(=O)Cc1cccs1)C2 N1(C(C2CC(=O)NC2)=O)CCCC(C(=O)Nc2cc(-n3cccn3)ccn2)CC1 c1(C(N2CCC(O)(c3ccccc3)CC2)=O)cc(=O)c2cc(C3CC3)ccc2o1 c1(C(N2CCC(O)(C(C)NC(CCCC#CC)=O)C2)=O)ncc(C#N)cc1C C1(CNC(C(C=C)(F)F)=O)CCC(O)CN1C(=O)Cc1c(C)noc1C N1(C(C2CCCN2C(c2ccsc2)=O)=O)CCCc2cc(F)cc(F)c21 N1(C(C(c2ccc(F)cc2)C)=O)CC2CCN(C(=O)C(F)(F)C(F)F)CCC2C1 CCCCC(=O)C(=O)N1CCCC(CCC(=O)N(C2CCCC2)CCO)C1 c1(CCC)nc(CNC(=O)CC2CCN(C(C)CNC3CCN(C)C3)C2)cs1 Cc1nccnc1-c1cn(CCC(N2CCN(CC3CC(CF)C3)CC2)=O)nn1 C(=O)(C1=NOC(C)C1)N1CC(NC(Cc2c(C)nccc2)=O)C1 C1(C)(CC)CCN1C(C1(NC(=O)C(C)SC)CCC1)=O CC(C)(C)C(O)Cc1cn(C2CN(C(=O)CCCN3CCCC(CO)C3)C2)nn1 C1(CCC(=O)N(C2CC(F)(F)C2)CC)(NC(C2CC2Cl)=O)CCCC1 C1(C(C)C)CCCN(C(=O)C(C)N(C(c2ccc(C#N)o2)=O)C2CC2)C1 c1(CC(N2CC(C(C)NC(C=CC)=O)OCC2)=O)c(CC)nn(C)c1CC C1(NC(c2cccc(=O)o2)=O)COC2(CCN(C(c3ccncc3Cl)=O)CC2)C1 C=CC1OCCC1NC(=NCC1CCCCC1)NCc1ccc(C)o1 C1(NC(C2CC(SC)C2)=O)CCCC1NC(=O)CNC(=O)OC(C)(C)C C12(NC(CCCC(C)=O)=O)CN(C(=O)CC3CC=CC3)CC1CS(=O)(=O)C2 N1(C(CC(C)(C)NC(C(C)CCN(C)C)=O)=O)CCC(O)C12CCC2 c1(C(N2CC3(CCC(CNC(CCC(=C)C)=O)O3)C2)=O)cc2cc(F)ccc2s1 Clc1cc(SCc2nc(-c3cnnc(Cl)c3Br)no2)ccc1I N12CCOC(C1)C2.c1(N(C(C)C)C(C2CCCO2)=O)cnn(Cc2cccnc2)c1 N1(C(C(C)NS(C)(=O)=O)=O)CCC(C)(CNC(=O)CNc2ccccc2)C1 N1(C(CCCSC)=O)CC(=O)NC2CN(C(c3ccc4nncn4c3)=O)CCC12 c1(C(=O)NC(C2CCN(C(=O)CC3C(C)(C)C3(C)C)C2)C)[nH]ncc1C#N C1(NC(C2CCC=CO2)=O)CN(C(=O)Cc2cccc(C(F)(F)F)c2)CCC1O N1(C(C(C)(C2CC2)OC)=O)CC2CN(C(=O)Cc3cccc(C)c3Cl)CC2C1 C#CC12CC(CN1C(=O)COC1CC(NC(C3CCCCC(=O)N3)=O)C1)C2 N1(C(Cc2n[nH]c(=NC)s2)=O)CC2(C1)CN(C(C1CCS1(=O)=O)=O)CCO2 c1(CC)[nH]nc(Cl)c1C(=O)NCC(C1CCCC1)NC(c1c(C)nsc1C)=O C1(NC(c2cc(OC)c(Cl)nc2)=O)CCCC2CN(C(=O)CC3(O)CCC3)CC12 C1(C(N2CCCC(COC)C2)=O)CC2CCC1N2C(=O)CCCn1cccc1 N1(C(CCc2c(C)noc2C)=O)CC2=C(C1)CN(C(=O)CC1CC3CC3C1)C2 c1(CCC(=O)NCCCC(C)NC(C(C)OCCC#C)=O)ccc(Cl)c(F)c1 CP(C)(=O)CC(=O)NCCC1(O)CN(C(C2(C3CC3)CCCO2)=O)C1 c1(C(N(C2CCC(NC(c3c(CCC)occ3)=O)C2)C)=O)ncn2c1CCC2 CC1(C)CC(CNC(=O)CCNC(N)=O)N(C(C2COC(=O)C2)=O)C1 N1(c2nccc(OCC)n2)CC(C)CN(C(C23CC(CO2)C3)=O)CC1C C1(CNC(C2(COC)CC2)=O)CCCCC1NC(=O)CCc1ncco1 c1(C(N2CCC(C(=O)OCCO)C2)C(=O)NCCCC)cnn(CCC)c1 N1(C(C(C)C)=O)CC2CCN(C(c3cnc(-c4ccccn4)s3)=O)CC2C1 c1(OC)cc(C(N2CC(NC(c3cnn(CCO)c3)=O)CC(C)C2)=O)cc(Cl)n1 C(=O)(C1Cc2ccccc21)NCC(C)(CNC(c1cc(C)cc(N)c1)=O)OC Cn1cc(C(N2CC(C)(C)C2c2ccco2)C(=O)NCCC2(C)CC2)ccc1=O N1(C(C(C)(CO)OC)=O)CCc2ccc(C(=O)NCCOC3CCC3)nc2C1 C(=O)(CC1CCC(=O)c2ccccc21)NCC(CN(C(C)=O)C)(C)C c1(C(=O)NCC=CCNC(c2noc(CC)c2C)=O)ccc(O)cc1[N+](=O)[O-] c1(C(N2C(CNC(CC3OCCC(OC)C3)=O)CC2)=O)cc(F)c(Cl)cc1Cl c1(CNC(c2cccc(CNC(=O)COCC)c2)=O)cncc(C(=O)NCC)c1 C(CCCCC(=O)NC(CCNC(c1nccc(C(F)F)n1)=O)C(C)C)OC CC1CC(O)CN(C(=O)C(CC(N)=O)NC(c2nc(=N)cc[nH]2)=O)C1 C12CCN(CC1)C(=O)NC(CO)CNC2=O.C(C)(C(=O)N(CC)CC)NC1CC1 c1(C(=O)NC2CC(C)(CNC(C(C)CC3CCC3)=O)C2)nn2cccnc2c1Cl C1(C(=O)N(CC=CCNC(C2(C(C)(F)F)CCC2)=O)C2CCC2)CCCCN1S(N)(=O)=O C(CCC)(C(O)C(=O)Nc1cccc(C(N)=O)c1)NC(CCC#CC)=O C#Cc1cc(F)c(C(=O)NCCCN(C)C(c2cncn2C)=O)c(F)c1 C1(NC(CCc2cnc(C)o2)=O)CCCC(NC(=O)CSCc2csc(=N)[nH]2)C1 C1(C(=O)NCc2cccs2)CN(Cc2cc(F)ccc2I)CCC1O c1(C(N2CC(NC(CC(=O)NC3CC3)=O)C2)=O)cc(F)cc2cccnc12 n1(CC)ncnc1C(N1CCCC1CCNC(c1cnc(N(C)C)s1)=O)=O CC1CCN(CCO)CCC1N(CC(=O)Nc1ccc(F)cc1)CC1CCNC1 c1(CC)cccnc1C(=O)NCC(C1CCN(C(c2nccn2C)=O)CC1)C C(C)(CO)(C(=O)NCCN(C(=O)CC1CCCO1)Cc1cccc(Cl)c1)OC Cc1c(C(=O)NC(C2(O)CCN(C(C3CN(C(N)=O)C3)=O)C2)C)cncc1F Cc1cc(C(=O)N(C(C)CN(C)C(c2cc(Cl)no2)=O)C)cc2nn[nH]c12 C=CCC(C(=O)N(CCC(=O)NCC(Cl)Cl)OC)OC N1(C(C#C)(C)C)CCN(C(C(=O)NC2CCCCC2)C(C)C2CCOCC2)CC1 N1(C(CCCN(C(=O)OCC)C)=O)CC(NC(c2ccc(C3CC3)o2)=O)C(F)C1 N1(C(COC2CC(NC(C(C)C3CCCC3)=O)C2)=O)CCCC2CNC(=O)C12 N1(C(C2CN(C(C)=O)C2)=O)CCCCC(NC(=O)C(C)(C)CCCF)CC1 C(=O)(CC(C)(C)CC)N(C1CCN(C(=O)CNC=O)C1)CCC C(=O)(C1=CC2(CCOC2)C1)N(C)CC1COCCN1c1ccnc(C(F)(F)F)n1 C1(NC(C(N)=O)=O)CCCCC1NC(=O)COCc1nc[nH]n1 C1(NC(c2ccc(CCC)[nH]2)=O)CCC2CN(C(=O)CC3CCC(O)C3)CC2C1 C1(C(N(CC(C)N(C(=O)CCOC2CC2)C)C)=O)CCc2c[nH]nc2C1 N1(C(CCOC)=O)CCC2CN(C(=O)CCNS(=O)(=O)c3cccs3)CC12 CC(C)C1=NOC(C(=O)NC2(CNC(=O)C(C)SC(F)(F)F)CC2)C1 c1(C(N2CCC(CN(C(C(CC)F)=O)C)C2)=O)cc(F)ccc1-c1ccccc1 CC1CCCCCC1NC(=O)NCC1CC(C(N)=O)=NO1 C1(C)(C(N2CC(N(C(CC3C(C)CCC3)=O)C)C2)=O)CCSCC1 C1(C(=O)NC23CC(CNC(C4CCC(C(C)C)CC4)=O)(C2)C3)CCCS(=O)(=O)N1 C1(NC(c2ccc(OCC)c(F)c2)=O)CCc2cc(OC)ccc2C1 C1(C(N2CC(=C)C2)=O)CN(C(=O)C(C)=C(C)CC)CCC1C C1(O)(C(=O)NCC(CC=C)NC(c2c(Cl)noc2C)=O)CCc2ccccc2C1 N1(C(C=Cc2n(CC)ncc2)=O)CCC2(CC1)CC2CNC(c1cncnc1)=O C(C1CCc2nccn21)NC(C1CC12CCN(C(c1cccc(O)c1F)=O)C2)=O C(=O)(C(C)(C)C(C)(F)F)N(C)CC1CN(C(c2cn(C)nc2C2CC2)=O)CCO1 c1(C(C)(C)NC(C2SCCS2)=O)ccc(-n2cc(CCS(C)(=O)=O)nn2)cc1 c1(OC)cc(C(=O)NCCCCNC(c2cnc[nH]2)=O)n(C)n1 CC(C)C(C)C(CNC(=O)C(c1ccccc1Cl)O)N=c1[nH]c(Cl)ncc1F N1(C(C)=O)CCC(C(=O)NCCOC2CN(C(=O)C(C)(C)c3csc(C)c3)C2)C1 C1(NC(C=CC)=O)CC(C(=O)OCc2nsc(CC)n2)C12CCOCC2 C1(C(C)C)CN(C(c2n[nH]cc2I)=O)CCN1C(=O)COC1CCOC1 CN=c1[nH]c(=NCCC(C)C)[nH]c(=NC2COc3ccccc3C2)[nH]1 C12CN(CCC1(F)F)C(=O)C2.c1(C(=O)NCCN)cnc(O)nc1O C(=O)(C1=CCC2CCC1N2C(=O)CCCc1cnn[nH]1)N(C(CSC)C)C C1(C(N2CCC(C)(NC(=O)CNC(c3ccco3)=O)C2)=O)CCC(N=[N+]=[N-])C1 CN1CC(NC(=O)CN2CCN(C(c3nc(Cl)cs3)=O)CC2)CC12CCC2 CN1CCCC(CNC(C2CN(C(C3CC(F)(F)C3)=O)CC2(F)F)=O)C1=O CC12COC(C(N3CCCC(NC(C4CC(CC5CC5)C4)=O)C3)=O)(C1)C2 CC1C(NC(C2CCCC(C(F)(F)F)O2)=O)CCN1C(=O)CCc1cnn[nH]1 c1(C(=O)NC2CCCC2CNC(C2(CO)CCCO2)=O)cncc(C2CC2)c1 Cc1cc(C(N2CC(C(C)(C)O)(CNC(=O)C3=CCC3)C2)=O)ccc1C1CC1 CCC(CC)C(F)C(=O)NCC1CCC(C(=O)NC2CC3CCC(C2)C3O)CC1 CN=c1cc(C(=O)NC(CCN(C)C(c2cn(C)c(O)n2)=O)C(C)(C)C)cc[nH]1 Cc1nn(C)cc1C(=O)N(C(CNC(c1nc(Br)c(C)s1)=O)C1CC1)C c1(C(N2CCC(O)(C(C)NC(=O)Cc3nncs3)C2)=O)ccc2scnc2c1 CC(C)CCC(=O)NCc1cnn(C)c1C(=O)NC1C(O)CC1O c1(N(CC(=O)NCC2(NC(=O)C(=O)N(C)C)CCOC2)C)ccc2cc[nH]c2c1 C1(N(C(COC)C)C)CC2CCC(C1)N2C(c1cncn(C)c1=O)=O c1(C(N(CCNC(C(C)=C2CC2)=O)C2CC2)=O)cnn2c(N)cc(C)nc12 N1(C(c2ccn(CCCC)n2)=O)CC2CCC(NC(=O)C=CC(C)C)(C2)C1 CCCC(CCCO)C(=O)NCC1CN(C(C2(COC)CCCO2)=O)CCC1C CCCCC(CC)CCC(=O)N1CCC(NC(=O)C(C)NC(=O)C2CC2)C1C N1(C(C(C)N2CCC2)=O)CC2CCC1C2NC(c1cc(C2CC2)n(C)n1)=O C(=O)(C(CC)(CC)CC(=O)OC)NC1C(NC(C2(C#C)CCCCC2)=O)C1 C(CC(CC)C(=O)NC(C)CCN(C)C(c1ccc(CNS(C)(=O)=O)o1)=O)=CC N1(C(C=CCC)=O)CCCC1C(=O)NC1CC=CCC1 c1(CC2N(C(C3CC(N=[N+]=[N-])C3)=O)CCCC2)nc2ccccc2s1 C#Cc1cc(C(=O)NCCC(C)(C)NC(c2ccc(F)cc2Br)=O)cc(F)c1 c1(C(N(C2CC(NC(CN(C(=O)OC)C)=O)C2)C)=O)[nH]c2ccc(F)cc2c1C C1(NC(C=CC(C)NC(=O)CN=[N+]=[N-])=O)CCCN(C)C1 C=CCC(CNC(=O)CC1COCCN1C(=O)CC1CCC(C)CC1)CC(C)C N1(C(C2CC=C(C)CC2)=O)CCC(C(=O)NCc2cccnc2F)CC1(C)C C1(C)(CCNC(C(CC)n2cncn2)=O)CCN(C(=O)CS(=O)(=O)NC)C1 CC(C)C(CNC(c1ccoc1Br)=O)NC(c1snnc1C1CC1)=O c1(C(c2n(CCOCC)nnn2)Nc2ccc(CCO)cc2)c(Cl)cccc1Cl c1(C(N2CCC(N(c3ncncc3C#N)C)C2)=O)cc(Cl)ccc1Br CC(C)CC(CC(=O)NC1CC(n2cccn2)C1)COc1cnn(C)c1 CC1C2CCC(C2)C1C(=O)NCC1=CCN(C(=O)CN2CCC(CO)CC2)CC1 c1(-c2cn(C)nc2)cncc(C(=O)NCC2(O)CCN(C(=O)CNC=O)C2)c1 N1(C(c2cncc(OC)c2)C(=O)NCCC(=O)OCC)CC2CCC2(C)C1 c1(C(N(CCC(C)NC(c2ccc(Cl)s2)=O)C)=O)ccc(C(F)F)nc1 n1(-c2ncc(C)cc2Br)ccc(=NC(=O)NCCc2ccccc2C(F)(F)F)[nH]1 N1(C(CC(CC)OC)=O)CCCCC12CN(C(=O)Cc1nc[nH]n1)C2 C=CC(CCC)CC(=O)NCC(CO)NC(=O)CCOc1ccccc1Br CC1=C(C(=O)N2CCCC(CO)(NC(=O)Cn3cc(N)cn3)C2)CCC1 C1(CNC(=O)Cc2sc(O)nc2O)CC(NC(c2n[nH]cc2Br)=O)C12CCC2 C(=O)(CC(C)(C)C(F)(F)F)NC(CNC(COCCCCC)=O)(C)C1CC1 n1(CCCOC)c(N2CCC(C)C2C(=O)OC)nnc1-c1ccc(Br)s1 Cc1nccc(Br)c1NC(C1CC1NC(c1ccccc1-c1cnco1)=O)=O C(CCCCCN=C(NCc1cccc(C(F)F)c1)NCc1ncnn1C)SC CCS(=O)CC(=O)NCc1csc(CNC(C2C3CC4C(C3)C24)=O)n1 CC(C)C(O)C(F)(F)C(=O)NCCCCCN(C)C(c1csc(C(N)=O)n1)=O CC(CC(=O)N1CC=CCC1C(N1CCC(F)(C(N)=O)C1)=O)C(C)(C)C C(CC(O)CNC(C1CCOC1C1CC1)=O)NC(C1(CC#C)CC1)=O C1(C(=O)Nc2c(OC)ncc(C)c2)CCC2CCC1N2C(C1OC2CCC1C2)=O O=[N+]([O-])c1cccc2c(NCc3cccc(OC(F)F)n3)ncnc12 C(CC(=O)N1CCC(C(N2CC(F)(C3CC3)C2)=O)O1)C1(C)N=N1 C(=O)(C(CC1CC1)NC(C1OCCC1CC)=O)OCC N1(C(c2cn(CC=C)nn2)=O)CC2CCOC2(CNC(=O)C(C)CS(C)(=O)=O)C1 N1(C(C)=O)CC2CCN(C(C3CCCSC3)=O)CC2C1 N1(C(CS(CC)=O)=O)CCC2CN(C(c3cc(=O)cc[nH]3)=O)CC2CC1 CC1CC2CN(C(=O)CCC#N)CC2N1C(c1ccc(CF)cc1)=O CC(C)(CCCNC(C1CC(O)C1)=O)NC(c1cccnc1N)=O N1(C(C2N(C)C(=O)NC2)=O)CCCC(C2CCCN(Cc3ccccc3)C2)C1 N1(C(C(=Cc2ccccc2)OC)=O)CC(C(=O)OC(C)(C)C)C(F)(F)C1 CCC(CN(C)C)CC(=O)NC(CCN(C)C)C(=O)NC1CC2(CCCC2)C1 N1(C(C(COC)O)=O)CCCCC1C1CN(C(=O)C(=O)NCCN(C)C)C1 C(=O)(C(C)(F)C(C)(C)F)NCCCC(C)NC(C(CC)CC)=O C1(C(F)(F)F)(C(=O)NCC2(OCC)CCOC2)CC2C=CC1CC2 n1(CC(=O)NCC2(OC)CN(C(C34CC(F)C3C4)=O)C2)nc(C)ccc1=O c1(CNC2C(C(=O)Nc3cnn(C)n3)CCC2)ccc2ccccc2n1 Cc1cncc(C=CC(=O)NC(C)(C)C(C)NC(=O)COC2CCC2)c1 C(=O)(CCN=c1[nH]ccs1)N1C2CC(NC(c3ccc(Cl)o3)=O)C1CC2 c1(OCC(C(=O)NC2C(NC(=O)CC3CC=CCC3)C2)O)ccccc1Cl Cc1nc(C)c(C(=O)N(C(C)CNC(=O)CS(=O)(=O)CC2CCCO2)C)nc1C CSC1=C(C(=O)N2CCCC2CNC(=O)C2=CCCC2C)CCCC1 c1(OC)cccc(OCC(=O)NC2CCC(CNC(C3(C)CCNC3=O)=O)C2)c1 c1(C(=O)NC(C)CN(C)C(C2CC3CCC2O3)=O)cc2sccc2cn1 c1(OC)ccc(Cl)c(C(=O)NC2(C)CCN(C(C3(SC)CC3)=O)C2)n1 C1(NC(c2cc(C(F)F)cs2)=O)CCCCN(C(=O)CCCCC2CC2)C1 C1(C(=O)NCC(CC(=O)NCC2CC(O)CCO2)OC)(CC)CC(C)(C)C1 Cc1[nH]c(C#N)cc1C(N1CCC(C)C1CNC(=O)C(=O)NCC1CC1)=O N1(C(c2cc(OC)ncc2)=O)CCCN(C(=O)C=Cc2ccc[nH]2)CC1 C(=O)(CCCCCn1cnnn1)N1C(C)CC(CNC(c2cnc(C#N)s2)=O)C1 Cc1ccc(CNC(=O)CC(C)NC(c2ccc(CO)nc2)=O)nn1 CCC1=C(C(=O)N(CC(C)CNC(c2sc3cccnc3c2Cl)=O)C)CCCO1 C(c1cnccn1)=CC(=O)Nc1cn(C2CCN(C(C(C)(O)C3CC3)=O)C2)nc1 C1(c2n(CCCC)nnn2)(NCC2OCCO2)COC2(CCCC2)C1 Cc1ncsc1CCC(=O)NC(C)(C)CCNC(=O)CCCn1ccnc1C C12(C(N3C(CNC(c4ccc(Br)cc4)=O)CCCC3)=O)CCCN1CC(O)C2 C1(OCC)CC(N(C)Cc2nc3ncccc3o2)C12CCCCC2 N1(C(CC(c2ccc(C)cc2)C)=O)CCN(C(C2CC(O)C2)=O)CC1CO C1(C(CNC(C(CC)NC(N)=O)=O)(C)O)CCN(C(=O)CSCC(N)=O)CC1 N1(C(C(=O)N(CC(C)O)CCN(C)C)=O)CC2CC3CC2C1C3 N1(C(C2N(C)CCCC2)=O)CCCC2CN(C(C3(F)CC=CC3)=O)CC12 C=C(C)CC(C(=O)Nc1cccc(C(C)C)c1)NC(=O)Cc1ccc(C)s1 C(CC(=O)N(C)Cc1ccncc1)(C(F)F)NC(c1c(CC)cc[nH]1)=O N1(C(C2(C)ON=C(C)C2)=O)CCN(C(c2c[nH]c(=O)cn2)=O)C(CF)C1 Cc1c(CCC(=O)NCC2COCC2NC(c2c(Cl)cnn2C)=O)cnn1C C=C(C)CC(C(=O)NCCC(O)CNC(c1csnn1)=O)NC(C)=O C1(NC(C(=O)Nc2c(C)n(C3CCOCC3)nc2)=O)CCn2c(cnc2C)C1 c1(C(N(CCNC(C2(COC(C)C)CC2)=O)C)=O)sc(Br)cc1Cl Cc1cn2c(n1)CCC(C(=O)NCC(C)CNC(c1cc(Cl)c(Cl)s1)=O)C2 N(C1c2ccccc2CCC1C)C(c1cc2c(cc1)C(NC(=O)OC)CC2)=O C(C(C(=O)NC(C(=O)NCC)C)NC(=O)C1CC1)OCC.C1(C)CS1 c1(CCN2CCC(N(C(=O)CCC3(C)CC3)C)C2)ccc(F)cc1F Cc1cc(C(=O)NC2CCCC23CN(C(C2C=CCCC2)=O)C3)cc(N)c1Cl C(=O)(CN=S(C)(C)=O)NCc1cn(C2CCN(C(c3sc(C)c(O)n3)=O)C2)nn1 C1(C(C)NC(Cc2c(C)occ2)=O)CCCN(C(c2ncccc2F)=O)C1 N1(C=O)CCCC(C)C1.c1(OC(C)C)cccc(SC(F)(F)F)n1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)N1CC(CC(C)NC(Cc2cn(CC)nc2)=O)C1 C1(C(=O)NC(C(C)NC(Cc2cncc(C)c2)=O)(C)C)Cc2cc(F)ccc2O1 C(C(CNC(=O)C=C1CCCC1)C(F)(F)F)NC(C1(NC(C)=O)CCCCC1)=O N1(C(C(C)SCCCC)=O)CCC(NC(c2ccc(Cl)s2)=O)C(CC)C1 c1(C(=O)OCC)ccc(S(=O)(=O)Oc2ccc([N+](=O)[O-])c(OC(C)C)c2)cc1F C(=O)(C(C)(C)CC#N)NC(CC)CNC(C1CC1OC(C)(C)C)=O CC1CCN(C(=O)CCc2ccncc2)C(C(N2CCCC(C#N)C2)=O)C1 c1(C(C)(C)C)nccc(=NC(=O)C2CC2C(=O)Nc2ccc(F)cc2C#N)[nH]1 N1(C(C(C)CS(C)=O)=O)CC2(CCN(C(C3CC3c3cccnc3)=O)CC2)C1 C1(NC(C2C(C)C2)=O)CC2CCC(C1C)N2C(=O)C(C)(O)Cc1ccccc1 C1(C)(COC)CC(NC(c2ccc(CO)cc2)=O)CN1C(=O)Cc1ccnn1C C1(CC(=O)NCCN(C(C(CC=C)OC)=O)CCCN(C)C)CCN(OC)CC1 c1(C(=O)NC(C)CCCNC(=O)CCNC(C2CCOCC2)=O)cccc(=O)o1 C=CCC(C(=C)C)C(=O)N1CC2(CCN2C(=O)C=Cc2cccc(Cl)c2)C1 c1(C(N2CC3C(C(=O)NC(c4ccccn4)C)C3C2)=O)cc(Br)nc(Br)c1 N1(C(=O)NCC)CCC(CN(C(C)CCNC(c2nc(CC)no2)=O)C)CC1 O(NC(=O)CN(C(=O)C=Cc1cc[nH]c1)CC)CC#C C(=O)(C(C)(C)C(O)C(C)C)NCC(C#CC(=O)NCCCCCOC)(C)C c1(C(N2CCC(C)(CNC(c3ccnc(F)c3F)=O)C2)=O)cc(Cl)cc(F)c1N c1(C(=O)NC2C(NC(=O)CCN3CCOC3=O)CCOC2)cc2ncccc2s1 Cc1sc(-c2cncc(C(F)(F)F)c2)nc1C(=O)NCc1cc(C#N)cs1 CCCCC(O)C(=O)NCC1CCC(NC(c2ccc(-c3ncon3)cc2)=O)C1 N1(CC(c2nnnn2C2CCOC2)NCc2cc(CC)on2)CCSC(C)(C)C1 C(N=c1[nH]c(=NCC2CC3CCC2C3)[nH]c2c1SCC2)c1c(C)nccc1 O=C1CS(=O)(=O)CC(C(=O)NCC2COCCN2C(=O)COC2CCOCC2)N1 c1(C(N2CCC(N(C(=O)C(F)F)CCC)C2)=O)sc(-c2ccccc2F)nc1C C(=O)(C(CC(F)F)N(C(=O)CCP(C)(C)=O)C)NC(CC)(C)COC CC(C)CC(C(=O)NCCc1ncccn1)ONC(C1(C)CNC(=O)C1)=O CCC(C(=O)N1CCOC(CNC(C2CN3CCCC2C3)=O)C1)C(C)C c1(C(N(C)C)=O)ccc(F)c(NC(c2csc(C3CCCO3)n2)=O)c1 C(=O)(C(F)CCC(C)C)NC(CCOCC)C(=O)NCC(C)CN(C)C N1(C(C(=O)NC(C)C)CC2(C#N)CC2)CCc2c(CO)n[nH]c2C1 c1(CC(C)NC(=O)CNC(c2ccnn2CC2CCCO2)=O)cc(Cl)ccc1Cl c1(C(C(=O)NCCC(CNC(C2(CC(C)C)CC2)=O)OC)F)cccc(C)c1 c1(OCCC)ccc(F)c(-c2ccc(NCc3ccncc3C(F)(F)F)cn2)c1 C1(CCNC(C(C)OCC(C)C)=O)CCCN(c2cc(-n3ccnc3)ncn2)C1 C1(C(=O)NCC2CC(O)(CNC(=O)CSc3nncs3)C2)(OC)CC(C)C1 C1(N(C(=O)C(F)=CCCF)CC)CCN(C(C2(N3CCOCC3)CC2)=O)CC1 N1(C(CCCOCCOC)=O)CC2CCN(C(=O)CN3CCC(C)C3)CC2C1 N1(C(C2(CC)CC2)=O)CCC(N(Cc2ccnn2C)CC2CC2)CC1 N1(C(c2ccc(C#C)nc2)=O)CCCC12CCCN(C(=O)C(C)C(C)C)C2 CCCCC(CC)CC(=O)NC(C)(CC)CCNC(=O)CC(CC)C(C)C c1(C(=O)NC2CC3(C(NC(C(N4CCNC4=O)C)=O)C3)C2)cncc2c1CCC2 C(CCN(C)C(c1cn(C)nn1)=O)(C(C)(C)C)NC(CC(CN(C)C)O)=O Cc1ccc(CN2CCOCC2C(=O)Nc2cnc(C)c(Br)c2)c(Cl)c1 c1(OC)ccc(NC(C2C3C(=O)OCC23Br)=O)cc1C#N C1(CC)CCN(C(=O)C(c2cnn(CC)c2)=O)C1CNC(C1(C(=O)NC)CC1)=O CCC(CC)CC(=O)N(CCNC(C1CNC(=O)CC1C(F)(F)F)=O)CC C1(CC)CCN(C(=O)CONC(c2ccc(CO)c(F)c2)=O)CCO1 N1(C(C2C(CC)C2)=O)CC2(CC2)CC1CNC(c1ccc(=O)n(CC)n1)=O C(=O)(CC1=CCOCC1)N1CCC(O)(CN(C(COC(CC)C)=O)C)C1 Cc1ccc(C(=O)NC2(C(=O)NCCC3CCCC(C)C3)CC2(C)C)cc1 C1(N(C(C(CC)=O)=O)C2CC2C)CCC2(CC1)CNC2 C1(C(N(C(C)(C)C)CC(N2CCC(C(C)(C)O)C2)=O)=O)CC(=O)CS1 c1(C(=O)NC2CCCC2C(=O)N(C)C)cccc(Cl)c1I.N12CCC(C(O)C1)C2=O S(=O)(=O)(c1cccc(=NCC2CCN(C(C)=O)C2)[nH]1)N(C1CC(=O)N(CO)C1)C CC1CN(C(c2cn(CCNC(C3(C(=O)N(C)C)CC3)=O)nn2)=O)CC(CO)O1 c1(C(=O)NC2CCC(CNC(CSC(C)C)=O)CC2)csc2ccncc12 c1(C(C)C)ccc(Br)cc1C(N1CCN(C(=O)C(C)C(C)(C)C)CC1)=O C(=O)(CC(F)(F)CS(C)(=O)=O)NCC(n1cc(CC2CCCOC2)nn1)C N1(C(c2ncccc2O)=O)CCN(C(=O)Cn2cncn2)C(CC(F)(F)F)C1 C(=O)(CC(CC)CC(F)(F)F)NC(CNC(CCCC#CC)=O)(CC)CC C12(CNC(C=CC(CC)C)=O)CCC(CC1)N(C(c1ccnc(OCC)c1)=O)C2 C1(C(=O)NCC2C(NC(c3cc[nH]n3)=O)C2)COCC2(CCC2)O1 n1(Cc2cn(CC3(C)CCCN3Cc3n(CC)ccn3)nn2)nc(C)c(C)c1C N1(C(c2ccc(C)cc2Cl)=O)CCC2CN(C(=O)C(C)Cc3cnn(C)c3)CC12 Cc1ncc(C(N2CCC(N(C)C(C3C4CC5C(C4)C35)=O)C2)=O)c(C2CC2)n1 C12(C(=O)NC(CC)CN(C(c3ccncc3Cl)=O)CC)CC3CC(C(=O)N1)C2C3 Cc1cccc2nc(C(N3CCC(NC(=O)CC(=O)NC4CC4)CC3C)=O)cn12 Cc1c(C(=O)NCC2CCN(C(C3CNC(=O)N3)=O)C2)sc2ccccc12 O=C(C1CCc2c[nH]nc21)NC1CCN(C(=O)CC23CCC(CC2)C3)CC1O c1(C(=O)NC2C(NC(Cc3ccn(CC)n3)=O)CCOC2)cc(C)cc(Cl)c1 N1(C(CSCC(N)=O)=O)CCC2CN(C(c3cccc4ncnn34)=O)CC12 c1(NC(c2c(OC)cccn2)C)cc(=NCC2OCCC2(C)C)[nH]cn1 c1(C(=O)NC2C=CC(CNC(CN(C3CCSC3)C)=O)C2)cc(Cl)nnc1O C1(NC(C2(C=C)CC2)=O)CCN(C(C2CCN2C2CCCC2)=O)CC(C)(C)C1 c1(CC)ccc(C(=O)NCC2COCC2NC(=O)C(F)(F)CC2CCCO2)nc1 n1(CCOC)ccc(C(=O)NCCC2CCC(NC(=O)CCc3nc[nH]n3)C2)n1 C1(NC(CCN(C)CC)=O)(CF)CCN(C(=O)C(c2cccc(Cl)c2)OC(C)=O)C1 c1(C(N(CCCN(C(=O)CCS(N)(=O)=O)C)C)=O)cccc(C(C)(C)C)c1N C(=O)(C(F)CC(CC)CC)NC(CCCC=C)C(=O)N(C)CC1(C)CCCO1 N1(C(C=CCC)=O)CCC(C2CCN(C(=O)CS(=O)(=O)CC(C)C)C2)CC1 CCC(CC(=O)N1CCC(C(N2CCC(OC3CC3)C2)=O)(CO)C1)C1CCC1 N1(C(C2(OC)CCN(C(c3c(COC)cco3)=O)C2)=O)CCCN(C2CC2)CC1 c1(C(=O)OC)cnc(NCC2CN(C(C3CC3F)=O)C2)c(Cl)c1 C(=O)(C(C(C)C)C(C)C)NC1(C(N2CC(COC)C2)=O)CCCC1C c1(C(=O)NC(CCN(C(CCC(C)SC)=O)C)C)nccc2[nH]nc(C(C)C)c12 N1(C(C(CC)SC)=O)CCCCC1C1(C(=O)NCC23CC(C2)C(C)O3)CC1 C1(NC(c2ccc3occc3c2)=O)CN(C(c2cc[n+]([O-])cc2)=O)CC(F)(F)C1 CC1OC2(C(=O)NCC3CCOCC3)CC1(NC(=O)CC1CCOC1)C2 C1(CC(=O)NCC2(SCC)CC2)(NC(C2CC(CN(C)C)CO2)=O)CCCC1 Cc1ccc2c(c1)C(=O)N(C(C)C(N1CCCC1CN(C)C(=O)C1CC1)=O)C2=O C1(CNC(c2[nH]cc(C)c2)=O)CCCC12CCN(C(=O)C1=CCOCC1)CC2 C1(NC(CNC(COC(C)=O)=O)=O)CC(NCCC2(C)N=N2)C1 c1(OC)ccc(NC(C2C3CCC(C3)C2NC(=O)CC=C(Cl)Cl)=O)cc1O N1(C(C2(c3cn(C)nc3)CCCO2)=O)C2CCC1CC(CNC(C1CSC1)=O)C2 C1(OC)CC(CNC(c2c[nH]ccc2=N)=O)N(C(=O)C=Cc2cscn2)C1 Cc1sc(Cl)nc1C(N1CCCCC1C(C)(C)CNC(=O)CC(C)(C)C)=O Cc1cnc(NC(C2CCCCN2Cc2c[nH]ccc2=N)=O)nc1 N1(C(c2cccc(OC)c2OC)=O)CC2CC(O)CC1C2.C(CCOC)OCC Cc1cc(C)c(C(N2CCC2CNC(=O)C(F)CC2CCCC2)=O)[nH]1 CS(=O)C=CC(=O)NCCC1(O)CCN(C(=O)CCCNS(C)(=O)=O)C1 c1(CNC(C(C)SC)=O)ccc2c(c1)CN(C(C1CCC(C(N)=O)C1)=O)C2 c1(OC)cc(C(N2CCCCCC2CNC(=O)Cn2ccnn2)=O)c(F)c(Cl)c1 C12(NC(C3(C=C)CCOCC3)=O)CCCN(C(C3CC4CCC(C3)S4)=O)CC1C2 c1(CN2CCC(NC(C(=O)Nc3ccc(C)cc3)C3CC3)C2)c(F)ccc(Cl)c1F c1(OC)nc(C)ccc1C(=O)NCC(F)CNC(c1ccccc1OC(C)C)=O c1(OC)cccc(C(CNC(C2(O)CCSC2)=O)NC(=O)CN(S(C)(=O)=O)C)c1 C(C1CCCCC1)=CC(N1CC(C(N2CCCC(OC3CC3)C2)=O)C(F)C1)=O Cc1cc(C#N)cc(C(=O)NCC2CCCN2C(C2(C)CCC(C)CC2)=O)n1 CCCC(CCCNC(=O)CN(C)C)NC(=O)CC1CN2CCN1CC2 c1(C(=O)NC(CN(C(=O)CC2OCCCO2)CC)=O)cc(C)cc(C)c1 C1(COC)(NC(c2cc(C)c(C)s2)=O)CCN(c2nnc(C)s2)CC1 N1(C(CC=CC=C)=O)CCC2(CCN(C(=O)C3CC3)CC2)C1 N1(C(C(CC#C)C)=O)CC2CN(C(C3CC(F)(CO)C3)=O)CCC12 C(C)(C)(C(C)CC(=O)NC1CCC1O)NC(c1c(C)cccn1)=O C(c1ccccc1)=C(COC)COC(=O)C(O)Cn1cncn1 c1(C(=O)NCC(CN(C(C2C3(CC3)C23CC3)=O)CC)(C)C)ccc(F)c(Cl)c1F Cc1ccc(C(=O)NC(CC2CCOCC2)C(=O)NC(C)CCC(C)C)c(F)c1 c1(NC(C2N(C(CC(CC)C)=O)CC(=O)C2)=O)cn(C)c(=O)nc1O C1(NC(CCSCCCC)=O)CC2(CCN(C(C3C4CC(=O)CC34)=O)CC2)C1 c1(OCC(N2CCC(N(C(C(CC)OC(C)=O)=O)C)C2)=O)c(F)cccc1F c1(C(=O)NCCCN(CCO)C(C2(F)CC2)=O)cccc([N+](=O)[O-])c1Br C=CC(O)C(=O)NC(C)(C(=O)NCC(F)Br)C1CCC1 C1(S(C)(=O)=O)(C(=O)NC2CCC(CCNC(CC3ON=C(C)C3)=O)C2)CCCC1 c1(C(=O)NC(CCOC)CNC(C2CCOCC2)=O)cnc(SC)n1C C(=O)(CC(C)CC(=O)NCC1CCC(NC(c2ncc(C)cc2F)=O)CC1)OC c1(C(=O)NCC2(C=C)CCC2)ccc(CNC(=O)CSC2CCCCO2)nc1 C(=O)(C1CCSc2ccccc21)N(C)CC1N(C(CCCCC(C)C)=O)CCC1 c1(OC)ccc(C(=O)NC(C)CNC(=O)C(c2ccc(F)cc2F)(F)F)c(F)n1 C1(C(C)NC(C2(C(=O)NC)CC2)=O)CCCN1C(C1CC(Cl)(Cl)C1)=O Cc1c(-n2cc(C3(O)CN(C(c4ncoc4Br)=O)C3)nn2)cccc1N Cc1ccc(C(F)C(=O)NCCC(O)CNC(=O)CN2CCCC2)cc1 Nc1c(C(N2CCC(NC(=O)C(F)C3CC3)C2)=O)ccc2c1CCCC2 C12(C(=O)NCCCCCCNC(c3n(C)cnc3)=O)CCOC1CS(=O)(=O)C2 C1(C)(C(N(CC(C)NC(=O)CC2CCC(=O)NC2=O)C)=O)CCN(C)CC1 CC(O)C(C(=O)NCCCC1CCCN1C(C1(C(N)=O)CC1)=O)NC(=O)C1CC1 Cc1ccc(C(N2CCCC2C(C)(C)CNC(C23CC(C)C2C3)=O)=O)c(Cl)c1 C1(O)(C(=O)NCC2CCN(C(C3(CC)CCOCC3)=O)C2)Cc2ccccc2C1 c1(C(=O)NCC(C(=O)N(CCCO)C)O)cccc(C(=O)N(C)C)c1 CC(CC(=O)NCC1CCCN1C(c1c[nH]c(C(N)=O)c1)=O)C1CCCO1 N1(C(C=CC2N(C)CCC2)=O)CCC(C)(C)C1CC(=O)NCCCN1CCCC1 C12(C(N(C(C)C)CCN(C(=O)C=CC3CC3)C)=O)CCCN(CC1)C2 Cc1ccc2c(C(N3C4CN(Cc5cc(F)ccc5Br)CC34)=O)cccc2c1 c1(OC)cncc(Br)c1C(=O)NCC1CCN1C(c1cc2scnc2[nH]1)=O C1(Cc2n(C)ncc2)CCCN(c2ccnc(NCc3cccc(Cl)n3)n2)C1 CN1CCOCC1C(N1CCCC1C1(C(N2CC(O)CC2CO)=O)CC1)=O N1(C(c2ccc(Br)s2)C(=O)NCCOC)CCc2ccc(CC(=O)OC)cc2C1 c1(C(=O)NCC2(O)CCN(C(CC3NC(=O)OC3)=O)C2)cccc([N+](=O)[O-])c1 C1(C(N(C2CC3CC3C2)C)=O)(CF)CCN(C(=O)CSC2CC2)C1 c1(C(=O)NCC(C(=O)Nc2cccnc2)OC)c[nH]c(C#N)c1C C(CCC(=O)N1CC(C2CC2)C1C1CC1)(C(C)C)NC(c1cc(=NC)[nH]cc1)=O C1(NC(c2nc(CS(C)(=O)=O)oc2)=O)CCCCN(C(=O)CC(C)(C)C#N)C1 c1(CC)nn[nH]c1C(=O)NC(C)(CNC(=O)C(Cc1ccccc1)OC)C1CC1 N1(C(c2ccc(CC)[nH]2)=O)CC2(CCC(NC(C3CC(C)C3)=O)CC2)C1 CN1CCN(C(C2(C)CCNC2=O)=O)CC1CNC(c1cc(C2CC2)n(C)n1)=O N1(C(C(CC)SC)=O)CCC(C)(C)C(C(N2C3CCC2CC3)=O)C1 N1(C(c2cc(C(CC)C)no2)=O)CCN(CC(C)NC(C2CCOC2C)=O)CC1 c1(OC)cccc(COCCC(N2CCN(C(=O)C=CCO)CC2)=O)c1 C#CC1(C(N2CC3CC3(CO)C2)=O)CCN(C(=O)Cn2cccc2)C1 c1(C(=O)NC(CCCC)CC(=O)O)coc2c(C(C)(C)C)cccc12 C1(CNC(C(C2CCN(C(C3(Cl)CCC3)=O)C2)C)=O)CCCCC1 C=C1CC2(C1)CC(C(=O)NC1CN(C(C3CCCCS3(=O)=O)=O)CCC1C)C2 C1(CC=C)(NC(=O)CCc2ccc(Cl)c(F)c2)CCCN(C(=O)C(C)CCCC)C1 C1(N(C(C(CC)SC)=O)C)CCCN(C(=O)CCC2CCCC2)CC1 C1(NC(c2cc(CC)[nH]n2)=O)CN(C(=O)C(O)C(C)(C)C)CC1N=[N+]=[N-] N1(C(C(C=C)CC)=O)CCC(C)N(C(c2ccc(C)cn2)=O)CC1 Cc1cncc(C=CC(N2CCN(C)CC2CNC(=O)C(C)C(C)(F)F)=O)c1 c1(CCC)sc(C(N2CCC2CNC(=O)CC2COC(CN)C2)=O)cc1CC N1(C(Cc2n[nH]c(=NC)s2)=O)CCC2CCCC(C1)N2C(c1ccc(C)nc1)=O C(=O)(C1CCCn2c(O)nnc21)N(C)Cc1c(F)cc(Cl)cc1Br C1(NC(C2CC=C(C)CC2)=O)CC(C(=O)NCCn2cncn2)=CC1O Cc1ccnc2nc(C(N3CCCC3CN(C)C(c3nncn3C)=O)=O)nn12 c1(CC(=O)NCC(CC=C)NC(=O)C(C)(C)C(=C)Cl)c[nH]c2ccc(C)cc12 c1(C(=O)NCCN(C(=O)CC2CCC2)CC)csc(N(c2ccccc2)C)n1 c1(C(CNC(c2cn(C)nc2)=O)NC(C2CCC3CC23)=O)cccc(Cl)c1Cl CC1(C(=O)N2CC(Cn3cc(CN(CCO)CCO)nn3)C2)CCCn2ccnc21 N1(C(CSC)=O)CCCC1CCNC(c1ccnn1C1CC1(F)F)=O c1(NC(C2CCC(C(=O)NO)CC2)=O)ccc2c(c1Cl)CCC2=O C(=O)(C(CC(C)C)C(C)C)NC(C(=O)N(CC(COCC)O)C)Cn1cncn1 N1(C(C(CC)C#N)=O)CCOC2(CCCN(C(c3cnn(C)c3SC)=O)C2)C1 C1(C)(C(N2C(CC(=O)N(C)CC3(O)CC(CF)C3)CC2)=O)CC(O)C1 c1(N2C(C)CN(C(C3CCCC34CC4)=O)CC(C)C2)nc2c(cc1Cl)C(=O)OC2 N1(C(CCOC(C)C)=O)CCC2(CC1)CN(C(C1CC1(Cl)Cl)=O)CC(C)O2 C1(NC(c2cc(CC)on2)=O)CC2CC1CN(C(=O)CC1(C)CCCC1)C2 c1(C(=O)NC2C(NC(C3C(C(C)C)C3)=O)COC2)ccc(Cl)cc1Br c1(CC(N2CC(N(C(=O)CCCNC(=O)OC(C)(C)C)C)C2)=O)ccc(F)cc1 N1(C(CCC(C)=O)=O)CC(C(N2CCCC(CO)C2)=O)C(C2CC2)C1 N1(C(C=Cc2ccc(SC)s2)=O)CC(C)CCC1CNC(=O)C(C)(C)C(N)=O CC1=C(C(=O)NC(C(=O)NC(C)CO)C2CCCC2)COCC1 Cc1cc(C(=O)NCC2CC2CC(=O)NCC2(N(C)C)CCOC2)c(N)s1 C1(CN(C(CC(=C)Br)=O)C)CCCN(C(c2cnc(O)o2)=O)C1 C1(C(N(C(C)CC(N)=O)C)=O)CC2(CCC2)CN1C(=O)CC1CSCCO1 C1(C(N2C(CNC(c3ccc(NC)cc3)=O)CCC2)=O)CCCC1C1CC1 c1(C(N(CCCNC(=O)C(C)C2CCOC2)C(C)C)=O)cnc2scnc2c1 c1(C(C)NC(c2cc(Br)ccc2Br)C)ccc2c(c1)OC(F)(F)O2 C(C(=O)NC(CN(C)C)C(C)C)(C(C)C)NC(C(n1ccc(C)n1)C)=O Cc1nn(C2CC2)cc1C(=O)NCC1(F)CC(NC(=O)CC#N)C1 C=C(C)C1OCCC1C(=O)N(C1(C(=O)N2CCCCO2)CC1)C C1(CCNC(C(C)OCC(F)(F)F)=O)CN(C(=O)Cc2cccnc2)CCCO1 C(=O)(C#CC1CC(F)(F)C1)N(C(CCNC(C(c1ccc(Cl)cc1)C)=O)C)C C1(NC(c2c(OC)c[nH]n2)=O)CN(C(C2CCC=CCCC2)=O)CC12CC2 C1(C(C)(C)CNC(C2CC=CCC2)=O)CCN(C(c2csc(C(F)F)c2)=O)CC1 C(C(CC(=O)NCC(=Cc1ccccc1)O)C1CCC1)NC(C=CCN(C)CC)=O c1(C(N2CC(CNC(C(=CC3CCCC3)C)=O)C(O)C2)=O)ccc2snnc2c1 C(CCC(=O)N1CCC(CN(C)C)C1)N(C(C=C(COC)C)=O)C N1(C(CC2(NC(C)=O)CC2)=O)C2CCC1CC(CNC(=O)C(C(C)C)C(C)C)C2 N1(C(c2n(COC)ncc2)C(=O)NCCSC)CCC(CO)C(O)C1 c1(SCCCC(N2CC(NC(C(C)OCC(F)(F)F)=O)C2)=O)cccc[n+]1[O-] N1(C(C(C)OC2CCOCC2)=O)CCC2(C1)CN(C(c1nccn1C)=O)CCO2 C(CC(C(=O)N1CC(C(O)C(=O)NCC2=CCCCC2)C1)OC)OC c1(C(N2C(CNC(CC3CC(=O)NCC3)=O)CCC2)=O)cc(F)cc(F)c1O c1(C(N2CC(NC(C(CC)CC)=O)C(O)CC2)=O)ccc2c(c1)OCO2 CC1=C(C(=O)NC2(C)CC(NC(C3CCN(C)CC3)=O)C2)Cn2ncnc2N1C c1(C(=O)NC2CCCCN(C(CCCC#N)=O)C2)c(Cl)oc2ccccc12 S(=O)(=O)(c1cnn2ccc(N3CC4CCC(F)(F)C4C3)nc12)N(CCCO)C CC1CCc2nc(C(=O)N(C)CCNC(C3CCC4(CCC4)O3)=O)cn2C1 CCC(O)C(C)C(=O)NC1CC(CNC(c2ccc(NS(=O)(=O)CC)nc2)=O)C1 CCCC(CCC)C(=O)N(C)CCN(C)C(c1cc(C)c(Br)s1)=O CCC(CC)(CC)C(=O)NCC1CCCCN1C(c1ccccc1SC(C)C)=O CC1OCCN(C(c2cnc(Cl)n2C)=O)C1C(=O)NCc1ccc(O)c(F)c1 C#CCC(C(=O)NCC(C)(CC)CO)NC(=O)CCC1CCCCC1 N1(C(C2C(C)C2)=O)CC2(CC(NC(c3cccc(Cl)c3C(F)(F)F)=O)C2)C1 N1(c2ccnc(C(C)C)n2)CCC2CC(C(N3CCCC(CO)C3)=O)C2C1 C1(CNC(C(CC)(C)OC)=O)CC2CCCC2N1C(c1ccnc(C(F)F)c1)=O Cc1cnc(C)c(C(=O)N(C)CC2CCN(C(=O)C=Cc3cncs3)C2)c1 CCC#CCCNC(C1(CNC(c2cc(C(C)C)[nH]n2)=O)CCCC1)=O CS(=O)(=O)CCCC(=O)NCCC12CCC1CN(C(c1ccc(C(N)=O)o1)=O)C2 c1(C(N(CCC)CCNC(C2CC2(F)Cl)=O)=O)cn(C(C)(C)C)nc1C(C)(C)C C1(CNC(=O)CCc2cnco2)CCC(C(N2CC(c3ncc[nH]3)C2)=O)C1 C=CCC(C)(C)C(=O)N(C)CC1(O)CCN(C(=O)CCN(C(CC)CC)C)CC1 C#CC1(NC(=O)C(F)(CNC(=O)CCn2ccnn2)C(C)C)CCC(C)(C)C1 N1(C(=O)OCC)CCC(C(C)NC(=O)C(=O)NCC2(C)CSCCO2)CC1 c1(C(C(=O)NCC(CC2CC2)OC)NC(C=CCCC)=O)cccnc1 c1(C(=O)NC2CC(NC(c3ccc(OCF)cc3)=O)C2)cc2cccc(Cl)c2[nH]1 C#CCC(C)(C(=O)NC1(CC(=O)OC)CC1)NC(=O)CCN=[N+]=[N-] c1(C(=O)NCCOCCCNC(Cc2nnc(C)o2)=O)cccn2c(O)nnc12 C1(CN(C(CCNC(C)=O)=O)C)CN(C(=O)CC2(C)CCCCC2)CCO1 N1(C(COC(C)=O)=O)CC2CC(NC(c3ccccn3)=O)CC(C2)C1 n1(C(C)C)cnc2c(N3CCOc4ncccc4C3)nc(N(C)C)nc12 n1(CCC)nc(-c2cccc(CC)c2)nc1-c1cnn(CN2CCCCC2)c1 c1(OCCCC)ccc(NC(=O)CCOc2ccccc2)cc1.C1(=O)CO1 N1(C(CNC(=O)OCC=C)=O)CCC(NC(c2cccnc2C)=O)CC1C1CC1 C1(C(C)(C)C)CC(C(=O)NC2CCC(C)N(C(c3cc4cscc4s3)=O)C2)=NO1 c1(C(N(CCN(C(C2(c3ncc[nH]3)CC2)=O)CC)CC)=O)ccccc1C c1(CNC(c2cnccn2)C)ccc(C2(C)CC2)cc1 CCC(O)C(C)C(=O)N1CCC(OCCNC(=O)Cn2cc(F)ccc2=O)CC1 Nc1cc(F)c(Br)cc1C(N1CC2CC1CN2C(C1(CCO)CC1)=O)=O N1(C(C2CC(C(=O)OC)C2)=O)CCCN(C(c2ccc[n+]([O-])c2)=O)C(C)C1 Cn1c(O)ncc(C(N2CCCC2COc2ccc(Br)cc2)=O)c1=O C(N=c1ccc(Br)c(S(=O)(=O)NCCc2ncccn2)[nH]1)c1n(C(C)C)ncn1 N1(C(C2CC(C#N)(OC)C2)=O)CCC2(CCCN(C(=O)Cc3nc[nH]n3)C2)C1 CON(CCC(=O)N1CC2(CCCCCC2)C1)C(=O)CCCC1CCCO1 N(C(=NCC1(CO)CCOC1)NC(C1CC1)C1CC1)C(CC=C)C CCCC(C)CC(=O)N1CCCC1CNC(c1ccc(CN2CCCC2)o1)=O C1(NC(C2C(C)CC2)=O)CC2(C1)CC2C(=O)NC(CO)C(=O)N(C)C O=C(CC1CCC(NC(C2(CCF)CC2)=O)C1)N=c1ccn(C(F)F)[nH]1 Cc1cnn2c1CN(C(c1n[nH]c3c1CN(C(C1CCC(F)C1)=O)C3)=O)CC2 N1(C(C2CCCC(OC)C2)=O)CCC(O)(CCNC(C2COC(=O)C2)=O)CC1 CC(C)C(O)CC(=O)N1CCCOC(CCNC(=O)Cc2ccccc2)C1 C1(C(N2CC(NC(CN(CC)CC)=O)C2)=O)(N(C)C)CCOCC1 Cc1ccc(F)c(C(=O)NC2CC3(C2)CC3NC(=O)C(O)C(C)C)c1Br c1(C(=O)NC2(C(N3CC(CO)CC3CO)=O)C(C)C2)cc(C#N)cs1 c1(C(CNC(=O)Cn2cc(Br)cn2)NC(C(C)N(C)C)=O)ccc2ccccc2c1 c1(C(C2CN(C(=O)C(C)NC(=O)OC)C2)C2CC2)cccc(F)c1OC CON1CC(C(=O)NCC(C)(O)CNC(c2nc(C)cs2)=O)CC1=O CC(C(=O)NCCOC1CCN(C(=O)CC2(C#N)CCC2)C1)C(C)O CC(CCCNC(=O)CCNC(c1ccccc1)=O)NC(=O)CC1CC1C1CC1 c1(C(N2CCC(OCCNC(c3cc(F)ccc3Cl)=O)C2)=O)cnc2n1CCS2 C(O)(CCNC(C1CCCC1c1ccncc1)=O)(C(F)(F)F)c1n(C)ccn1 N1(C(CCC(=O)OCC)=O)CCCC(NC(C2(C)CC3(CCC3)C2)=O)CC1 C1(CNC(c2nc(C)n(C)n2)=O)CN(C(=O)C2=CC(C)(C)C2)CCC1C CC(C)C(O)C(C)(C)CN=c1[nH]c(=NCCS(=O)(=O)NC2CC2)c2ncccc2[nH]1 c1(NC(C2(F)CCN(C(C(OC)OC)=O)C2)=O)cc(C)c(F)c(C)c1 CCC(C)(C)C(=O)C(=O)NCCCN(CCO)C(C1CCCC(C)(C)CC1)=O c1(C(N2CCC(CCN(C(C(CC3CC3)OC)=O)C)CC2)=O)ccnc(C)c1N C1(NC(CNC(c2ccc(C)cc2)=O)=O)CCCCN(C(C2(CO)CCC2)=O)C1 Cc1c(Cl)cccc1S(=O)(=O)NC1CCOC(C)C1C C1(NC(C(C)NC(CC)=O)=O)CC12CCN(C(=O)CCCS(N)(=O)=O)CC2 C(=O)(C1=CC2(CCOC2)C1)N1CC(NC(=O)C(CO)C(F)(F)F)C2(CC1)CC2 C1(CNC(CSc2ccc(C)cc2)=O)CCN(C(=O)C(F)(F)C(F)F)CC1C C1(CNC(C2(CCC=C)CC2)=O)CC2CCC(C1)N2C(c1cccc(F)c1F)=O N1(C(COC2CC(NC(C3N(CC)CCOC3)=O)C2)=O)CC2(CC2)CC1C CCS(=O)(=O)Cc1cn(CCC(=O)NCCCOC2CCC2)nn1 CC1CC(CNC(C2CC3(CC3)C2)=O)CN1C(=O)C(C)CN(C)C Cc1csc2c(N3CC4CCC3CN4Cc3ccc(F)cc3)ncnc12 O=C(C1CCCc2ccccc21)NCCNC(C1(C(F)(F)F)CC2CCC1C2)=O C1(C(N2CC(OCCC(=O)NCCNS(C)(=O)=O)C2)=O)CC2CC(=O)C1O2 c1(C2(CNCCc3onc(CSC)n3)CC2)ccc(C=CC(=O)O)cc1 c1(C(N2CCC(C)C2CNC(c2cc(=O)cc[nH]2)=O)=O)cc(O)ccc1O N1(C(C(C)C(C)(F)F)=O)CCN(C(c2nnc(O)cc2O)=O)CC(CO)C1 N1(C(C2(SC)CC2)=O)CC(C)C(C)(CNC(=O)CC2CSCCO2)C1 c1(C(N(CCC(N2CCC(OCC3CC3)C2)=O)CC)=O)nnccc1C O=C1NC(=O)C2(CN(C(c3cccnc3OCC(F)(F)F)=O)C2)N1 c1(C(=O)NCC2(O)CN(C(c3c(CC)occ3)=O)C2)cc2scc(C)c2[nH]1 C=CCC(CC=C)C(=O)N1CC2(CCCC2NC(=O)C(O)Cc2cnn(C)c2)C1 c1(CN2CCCC(C(N)=O)C2)ccc([N+](=O)[O-])cn1.N12C3CCC1C(C3)C2=O C(CCCCC(=O)NC1(C)CC(NC(=O)CC23COCC(C2)C3)C1)OCC c1(C(N2CC(NC(C=C(CC)CC)=O)C(C(F)F)C2)=O)[nH]c(C)c(C(C)=O)c1C C1(c2nc(-c3ccc(OC)cn3)nn2CCC2CC2)CC12CCSCC2 N1(C(C2CCC(N(C)C)C2)=O)CC2CC2C1CNC(c1ccn(C(F)F)n1)=O N1(C(CCSC)C(=O)NC(C)(C)C)CCOc2ccc(C(C)C)cc2C1 Cc1ccc2c(Cl)c(C(N3CCC(CN(C(=O)C(C)CF)C)CC3)=O)sc2c1 c1(CC(=O)NCCC2CCN(C(COCCC)=O)CC2)ccc(F)c(OC)c1 C(=O)(C(O)C(F)(F)F)NC(C1CCCN1C(c1ccc(=O)n(C2CC2)c1)=O)(C)C Cn1ncc2ccc(C(=O)NC3C4CC3N(C(C3(C)CCCCC3)=O)C4)cc12 CC(CS(C)=O)C(=O)N1CC(n2cc(CN3CCC(N)CC3)nn2)C1 CC1Cc2c(Cl)cccc2C1NC(=O)C(=O)Nc1cccc2c1OCC(=O)N2 N1(C(CC(C)(C)C2CC2)=O)CCCC2(NC(=O)C(C3CCOCC3)O)CCCC12 CCCCC(CCCC)N1CCC(NC(C)CC(C)(C)C)CC1 CCC(C)CC(C)N(C)C(c1ccoc1CNC(c1cnn(CCO)c1)=O)=O Cc1cncc(C=CC(=O)NC2CC2NC(c2coc3c2COC3)=O)c1 c1(CS(N2CC(C)=C(C)C2)(=O)=O)ccc(Cl)nc1C(F)(F)F N1(C(C2C(CC(C)C)C2)=O)CCCC(O)(CN(C(=O)Cc2ccc(CC)s2)C)C1 C1(C(NOCC)=O)CCC(C)(C)N(C(c2[nH]cc(C)c2C)=O)C1 C1(C(=O)OC)CN(C(c2cccc(F)n2)C(=O)NC2CCOC2)CCO1 CC(C)CC(C)(CNC(c1cc(O)nc(C2CC2)n1)=O)NC(C1CC1(C)C)=O c1(C(=O)NC2CC(C)(C)N(C(C3C(C)(C)C3(C)C)=O)C2)ccc(Cl)c2occc12 N1(C(C2(C)CCC(C)CC2)=O)CCOCC(C)(CNC(=O)COC(F)(F)F)C1 C1(CCC)(NC(=O)C(C)OC)CCCN(C(c2ccc(N)cc2OC)=O)C1 c1(C(=O)NC2CCCC(NC(C3CC(O)(CC#C)C3)=O)C2)c(F)ccc(F)c1O C1(CNC(CCC=C)=O)C2CN(C(=O)CC(CC)NC(=O)OC(C)(C)C)CC12 C1(CCC)CC(C(=O)Nc2csnc2-c2ccccc2)CCO1 c1(C(N2CC(C)(NC(C3COCCO3)=O)C2)=O)ncc(Cl)cc1F c1(Cc2scc(C(=O)NCC(CNC(C(C)(O)C3CC3)=O)F)n2)ccc(F)cc1 C(=O)(CCN(C(=O)CN(C)C1CC1)C(C)C)NCCOC1(OC(C)=O)CC1 c1(C(=O)NC(C(=O)N2C(COC)CC2)Cc2cc[nH]n2)cn(C)cc1C C12(C(=O)NCCCn3cc(-c4c[nH]nc4F)nn3)CC3CC(C(=O)N1)C2C3 N1(C(Cc2c(C)nc[nH]2)=O)CCC2(CCCCC2NC(C2CC2C2CC2)=O)C1 Cc1cc(C(=O)NC(CN=[N+]=[N-])C(=O)NC2CCC(=O)NC2C)cc(C#N)c1 C1(C)(C(=O)NC(CC(C)C)CNC(=O)Cc2ccc(Cl)s2)CC2(CCC2)C1 c1(C(C(=O)NCC=C)N(C2CCN(S(C)(=O)=O)C2)C)ccc(OCC)cc1C C1(O)(CNC(=O)CN2CCCC2=O)CCN(C(C2(CC3CCC3)CC2)=O)C1 CCCCC(C)CCC(=O)NCC(=O)NCC(=O)N(CC(C)(C)O)C CCC(O)CS(C)(=O)=O.C(=O)(CC)NC.N1(CCOCCO)CC1 C1(CC(C)C)C(=O)N1C(c1ccc(N)cc1)=O.C(C)(C)(C)OC(C)=O CC1c2ccccc2OC1CC(=O)N(C)CCNC(C12CCCC(CO1)C2)=O C#Cc1ccnc(C(=O)NC2CCCCC2NC(=O)CCNC(=O)CO)c1 C(C)(CC(C)(C)OC)NC(C(C)N(C(C(C)=CCC)=O)CC1CC1)=O N1(C(C2N(C(C3CC(OC)C3)=O)CCOC2C)=O)CCn2c(C)nnc2C1 c1(OC)ccc2occ(C(=O)NCC(CO)NC(C3CCC(O)CC3)=O)c2c1 C1(NC(CCCn2c(C)cc(C)n2)=O)CCCN(C(c2cnc(S)[nH]2)=O)C1C C1(CC)CN(C(=O)CC2(C)CCCO2)CCN1C(=O)COc1cccnc1 c1(CC)ccc(C(=O)NC2(CNC(c3c(C)nsc3NC)=O)CCCC2)nc1 C1(NC(C2N(C(c3c(NC)cnnc3)=O)CSC2)=O)CC(O)CC(C)(C)C1 C1(C(=O)OC)CCCCC1C(=O)NCCCCCCN(C)C(C1CC2CC2C1)=O c1(C(=O)NC(CC(C)NC(c2c(OC)scc2)=O)C)cc(S(N)(=O)=O)c(Cl)o1 C(=O)(C(OC)OC)N(CC(=O)NC(C1CCOC1)C#C)C1CC1 CC1=CCC(C(N2CC(O)(C(C)NC(=O)CCc3cnn(C)c3)C2)=O)CC1 c1(C(=O)NCC(C(C)C)(C)NC(C2CC(C)(C)C2)=O)n[nH]c2c1CS(=O)(=O)CC2 C=CCC(C)N=c1[nH]c2c(c(=NCc3ncc(Br)cc3F)[nH]1)CC(C)CC2 C1(CNC(c2onc(CC)c2C)=O)CCN(C(C2CCC(C)CC2)=O)CC1(F)F C(=O)(CCCCC(=O)NCc1ccccc1CNC(=O)C(C)(F)C(F)(F)F)NC c1(OCC)ccc(OC)cc1CN1CCC2CCCC12 N1(C(C2N(C)C(=O)NC2)=O)CCC2(CCCN(C(c3cnncc3O)=O)C2)C1 CC(C)C(CC(=O)NC1CC1c1ccsc1)NC(c1ccnnc1)=O CC1CN(C(=O)Cc2cc(C(F)(F)F)co2)CCC1CNC(=O)C(C)(Cl)Cl C(CC(O)C(=O)NCC(C)N(C)C(C1CCCC1(C)C)=O)SC C1(CC)C(=O)N(C)CCN1Cc1cn(-c2cc(Br)ccc2OC)nn1 N1(C(c2c(CC)c(C)ccc2)=O)CCC2(CC(NC(C3(C)CCCN3C)=O)C2)C1 c1(CC(N2CCC(N(C(C3CC(N(C)CC)C3)=O)CC)C2)=O)ccc(F)c(C)c1 c1(C(N2CCC(F)(CNC(C(C)n3cccc3)=O)CC2)=O)ncsc1S(N)(=O)=O c1(C(=O)NC2CCC(NC(c3csc(Cl)n3)=O)C2)cc(F)ccc1Br c1(C(=O)NCc2ccc(CNC(C34CC(F)C3C4)=O)cc2)ccc2nonc2c1 C1(C(=O)NC2CCCN(C(Cc3nc(C)c(C)s3)=O)C2)CCCC(F)(F)C1 c1(C(=O)NCCC(CNC(C2C(C)(C(C)C)C2)=O)(C)C)cc2ccncc2s1 S(=O)(=O)(c1cccc(C(=O)NC2CC2CNC(=O)C#CC(C)(C)O)c1)NCC#C c1(C=O)ccc(F)c(C(=O)NCCC2CCOC2)c1.C(CNC(C)C)OC c1(C(=O)NC(CC)CNC(C2(COC)CC=CCC2)=O)cc2ccccc2o1 c1(C(=O)NC2C(CNC(c3ccc(Cl)cn3)=O)CC2)cc2ccncc2s1 C1(NC(CCCC=C)=O)CCC2CCN(C(=O)CSc3nccn3C)C12 CC(C)CC(C(=O)NC1C(=O)OCC1(C)C)ONC(=O)C(O)Cn1cncn1 c1(C(=O)NC2CC3CC(NC(c4c(C)n[nH]c4)=O)C2C3)cc(C)c2[nH]cnc2c1 C(=O)(CCCC(C)(C)N1CCC(c2noc3c2CCCC3)CC1)NCCOC C(=O)(C(C(C)C)OC)NC(C(=O)NCC(C(=O)NCC)C)(C)C1CCC1 CC12CCC(CNC(=O)C(=O)N3CCCC3)(CO1)C2 c1(NC(=O)NCc2cccc(C3CCC3)c2)ccnc(Br)c1 c1(CC(=O)N(CCC(C)NC(=O)CCc2cn(C)cn2)C)csc2nccn12 C1(O)(CNC(c2c(C(C)NC(C3CC(N(C)C)C3)=O)noc2)=O)CCCC1(C)C c1(C(=O)OCC)csc(CN(C2CCN(C(=O)CC3CCOC3)C2)C)n1 C(C1CC(=O)Nc2ccccc21)NC(N1CCN(C(C2CCCC2)C)CC1)=O Cc1ccc(C(=O)NCC(C)NC(c2cc(C(N)=O)c[nH]2)=O)c(F)c1Cl CCCCC(CC)CC(=O)NCc1nocc1C(=O)N(CC(C)C(C)C)C c1(C2(C(N3CCC(c4nn[nH]n4)(C(F)F)C3)=O)CC2)ccc(Cl)c(Cl)c1 n1(-c2c(CNC3=NCCN(CCC)CC3)cccc2)nc2ccccn2c1=O C1(C(=O)NCC2(CC(C3CN(C)C3)=O)CCC2)CCN(OC)C(C)(C)C1 C1(N(C(C2(C3CC3)CCCO2)=O)CC)CCCN(C(=O)CC2CN(C)C2)CC1 C1(NC(c2cc(CNC(C3C(C(N)=O)COC3)=O)on2)=O)CCC(CO)CC1 N1(C(c2c(CNC(C=NOC)=O)ccs2)=O)CCC(OC)C1(C)C C1(NC(C23C(C)OC(CC2)C3)=O)CCN(C(C23CCC(C2)OC3C)=O)CC(O)C1 N1(C(C2CCC(N(C)C)CC2)=O)CC2=C(C1)CN(C(c1ccc(Cl)cc1N)=O)C2 c1(-c2nc(C)c(C(N3CCC(O)C3)=O)cc2)c(F)c(F)c(O)c(F)c1F N1(C(CCC(C)C)=O)CC2CCCC(Nc3cc(Cl)ncn3)C2C1 c1(COC)cccc(CC(=O)NC2CCCC2NC(=O)Cn2cc(Cl)c(C)n2)c1 CC1CN(C(=O)CC2C=CS(=O)(=O)C2)CCCN1C(c1cc(C#N)ccc1O)=O C1(CCONC(c2ccnn2CCO)=O)CCCNC1C(F)(F)F N1(C(C(C=C=C)C)=O)CCN(C(c2c(Cl)csc2Cl)=O)CCC1C N1(C(CCC=C(C)C)=O)CC(N(C2CC2)C(=O)OC(C)(C)C)CC1C1CCCC1 c1(OC)ccc([N+](=O)[O-])c(NCCC(C)(C)NC(c2nc(Cl)sc2C)=O)n1 N1(C(CCC#CC)=O)CC2(C1)SCCC2NC(=O)CCc1ccc(C)c(C)c1 C=Cn1nncc1C(=O)NC1C2CN(C(=O)C(C)Sc3nnnn3C3CC3)CC12 C1(NC(=O)C(c2ccccc2)F)CCCCN(C(C2(Cl)CC2)=O)C1 c1(C(=O)N(CCN2CCCC2c2ccsc2)C2CC2)ncc(C(F)(F)F)[nH]1 Cc1cc([N+](=O)[O-])ccc1-n1cc(C2CCN2C(=O)OC(C)(C)C)nn1 C(=O)(C(C)C(C)(C)C)NCCCC1(NC(C(c2ccc(F)cc2)OC)=O)CC1 N1(CC(=O)NC2CCCC2NC(C2(CCNSC)CCCC2)=O)CC2CCC1C2 c1(OC)ccc(CC(N2CCCC(NC(=O)C(F)C3CCC3)C2)=O)cc1F.C(=O)OC N1(c2ncn(C)c(=O)c2Br)CCC2CC(NC(=O)CCCN=[N+]=[N-])CCC2C1 C1(C(=O)N(CC(C2CCCC2)O)C)(CC)CCCN(C(=O)C2=NOC(C)C2)C1 N1(C(CCc2ccc(C)cn2)=O)CCN(C(=O)C(C)CC2CCCC2)C(C)C1 c1(CCCC(N2CCC(O)(CC(C)C)CC2)=O)c[nH]c2cc(Cl)ccc12 n1(C(CC)C)nc(-c2ccncc2)nc1C1CCc2cc(Br)ccc21 CC1=C(C(=O)N2CC3CC(C(N4CC(O)CCC4C)=O)(C3)C2)CCO1 C1(CC(=O)NC2(CN(C)C(c3ccnc(F)c3O)=O)CC2)CCCNC(=O)C1 CC(C)C(O)CC(=O)N1CCC(CNC(=O)C=CCN2CCCC2)C12CC2 CN1CCC(n2nc(CCN(C)C)nc2-c2ccccc2-n2cnnn2)CC1 Cc1nccnc1C(=O)NCC1CCN1C(=O)COC1CCCC(C)C1 CC(O)CCCC(=O)N1CCN(c2cc(C(=O)NC3CC34CCC4)ccn2)CC1 C1(CC(=O)NC2(CO)CCN(C(C(C)CN(C)C)=O)C2)CC(=O)NC(=O)C1 CN1CC=C(C(=O)NCC2(O)CN(C(=O)COc3ccccc3F)C2)C1 C1(N(C(COC(CC)C)=O)C)CCC(NC(c2ccnnc2NC)=O)CC1 c1(NC(C2CC(NC(C3CC(=O)NC3)=O)C2)=O)ccc(C(F)F)c(F)c1 n1(CC(N2C(C3(NC(C(CCC)O)=O)CC3)CCC2)=O)ccc(=O)cc1C N1(C(CCCNC(C)=O)=O)CC(C)CCC1CNC(c1cc(C)ccc1Br)=O C12(C(=O)NCC(C(C)C)(C)NC(c3ccc(C#N)cn3)=O)CCCN(CCC1)C2 C1(NC(CC2N(C(C(C)C3CCC3)=O)CC(O)C2)=O)CCCCCC1C N1(C(C2ON=C(C)C2C)=O)CCN(C(C2CC(C)C2)=O)CC12CC2 c1(C(=O)NC(C)CCNC(=O)CSC2CC2)cc(C(F)(F)F)ncn1 C(N=c1[nH]c(=NCCC(C)CO)c2cccc(F)c2[nH]1)c1cc(C)nc(O)c1 Nc1cc(C(N2CCCCC2CNC(=O)C(F)(F)c2cccnc2)=O)ncc1F CC(C)CCCC(=O)N1CC2CC1C2NC(c1cn(C)nc1OCC(F)(F)F)=O c1(C(=O)OC)cnn2c1CC(NC(=O)Cc1ccc3ccoc3c1)CC2 CCCCCC(C)CC(=O)NC(C1CN(C(C2CCn3c(O)nnc3C2)=O)C1)C N1(C(Cc2c(C)nc[nH]2)=O)C2CCC1CC(CCNC(C1(F)CCCOC1)=O)C2 C(=O)(C1=C(C#N)CCC1)N(CCC(N1CCC(CN(C)C)C1)=O)CCCO C(=O)(CC(C)CC(=O)NC(C)Cn1cc(-c2cscn2)nn1)OC Cc1oc(C#N)cc1C(N1CC(C(=O)NCCC2(CO)CC2)CCC1C)=O S(=O)(=O)(c1ccc(C2CC2Br)cc1)NCC1C(NC(C(C)C)=O)CCC1 C1(N(CC)CC)CCN(c2nnnn2C2CC(NC(C)=O)C2)CC1 C(=O)(C1=COCCO1)NC(C(C)NC(=O)CCN(c1ccccc1Cl)S(C)(=O)=O)C n1(CCC(=O)NC(C)CCN(C)C(c2ocnc2C2CC2)=O)cc[nH]c(=O)c1=O c1(CNC(C(CCCC)O)=O)cnn2c1CN(C(c1cnn(C(C)C)n1)=O)CC2 C1(C(C)(C)O)(CNC(=O)C=CCO)CN(C(=O)Cn2nnc(=N)[nH]2)C1 C#CC(CC1CCCCCC1)N=c1[nH]c(OC)cc2nccn12 N1(C(CS(CCC)(=O)=O)=O)CCCC2(NC(c3cnco3)=O)CCCC12 c1(C(=O)NCC(CO)NC(c2cnc(C(C)C)s2)=O)cc(O)cc(F)c1 Cc1ccsc1C(=O)NC(C)(C)COCCCNC(=O)CN1CC2CC2C1 C(C1c2ccccc2CN1C(=O)C(C1CCOCC1)F)NC(CCNC(C)=O)=O CCC(C)(C(=O)N1CCCC(CN(C(=O)CCCC2CC2)C)C1)OC C1(COC)(CNC(=O)C(C(C)C)NC=O)CCN(C(=O)CSc2nncs2)CC1 C1(C(=O)NCCCCNC(C2(OC)CCSC2)=O)CS(=O)(=O)CN1C(C)=O C1(N(C(CC=CCNC(COCCCOC)=O)=O)C)CCC(C)C1 c1(NC(c2n(CC)ccn2)=O)ccc(NC(C2CC=CCO2)=O)cc1C N1(C(CC(c2ccc(OC)cc2)C)=O)CCN(C(=O)C=C(C)Cl)CC1C1CCC1 C12(C(N(CC#C)C(C)C)=O)CC(C)(CN1C(C1CC(=O)CCO1)=O)C2 C(C(CNC(c1n[nH]cc1[N+](=O)[O-])=O)C(F)(F)F)NC(C1(C)CCOC1)=O c1(CC(=O)N(C)CC2CCN(C(=O)C(N)=O)C2)cc(C(F)(F)F)n(C)n1 C1(NC(CNC(c2cc(C)nn2C)=O)=O)CC2CC(NC(C3CCSC3)=O)C1C2 c1(CC)c(OC)cccc1CNC(=O)CCCC1(C)N=N1.C12(CC1)CC(=O)NC2 C12(CCC3C4C=CC(C4)C13)C(C(=O)OC)N2.c1ccccc1OC.c1ccsc1 N1(C(C2C(C(C)NC(c3c(C)n[nH]c3)=O)C2)=O)CC(CO)C(C)(C)C1 C1(C(N(CC(c2ccccc2)O)C)=O)CN(C(C2(Br)CC2)=O)CCN1 c1(C(=O)NCC2(OC)CN(C(c3c(OC)ccnc3)=O)C2)ccnc(C#N)c1 c1(C(=O)NC2(CC)CCN(C(CCOCC#C)=O)CC2)cc(C)c(N)c(C)c1 c1(CNC(c2cccnc2)C)cn(CCO)c(=O)nc1O N1(C(=O)NCCCSC2CC2C2CC2)CC2(CO)CCCC2(CO)C1 N1(C(Cn2c(C)cc(C)n2)=O)CC2CC(C1)CN(C(=O)C(C#N)C1CC1)C2 c1(N(C(C(CC)Oc2ccccc2Cl)=O)C)cccc2cc[nH]c12 C1(NC(C=CS(C)=O)=O)CN(C(c2ncc(C(N)=O)cc2Cl)=O)C2(CCC2)C1 C1(CNC(=O)Cc2cscn2)COCCN1C(=O)COCC1CCCOC1 C1(C(N2CCCC2CNC(=O)CCn2ncn(C)c2=O)=O)(OC)CCC12CCC2 C(C(N=c1[nH]c(Cl)c(C#N)s1)c1ccccc1)NC(C(C)SC)=O CC1(CC(=O)NCCOC2CN(C(=O)CC3CSCCS3)C2)CCS(=O)(=O)N1 CC(CNC(=O)Cc1ccccc1)C(=O)NC1CN(C(=O)C(C)C2CCCO2)C1 N1(c2n(Cc3c(OC)nc(C)cc3C)c(C3CCC3)nn2)CCNC(=O)C1(C)C c1(-n2c(C3(c4ccncc4)CC3)nc(C(CCC)C)n2)ccc2nc(C)[nH]c2c1 CC1CCC(C(=O)N(C)CC2(O)CN(C(C3CN(C)C3)=O)C2)S1 c1(NC(COCCNC(c2n(CC)c(O)nc2)=O)=O)ccc(C)cc1C CC(C)C(O)C(=O)N1CCN(c2cc(CNC(=O)CO)ccn2)CC1 Cc1c(C(N2CCSC(NC(CCNC(C)(C)C)=O)C2)=O)ccc(F)c1F N1(C(C2C(C(N)=O)C2)=O)CC(NC(=O)CSCc2ccc(Cl)s2)CC(F)C1 C1(O)(CNC(C(C)(C)NC(=O)NCCC)=O)CCN(C(=O)C(O)C(C)(C)C)CC1 c1(CC(=O)N(CC(C)(C)CNC(C2CC23CCCC3)=O)C)cccc2cn[nH]c12 C1(C(=O)NC2CN(C(=O)CC3CC(C)(C)C3)CC2C)(OC)CCOCC1 CCC(CN(C)C)CC(=O)NC(c1ccc(Cl)c(I)c1)CC c1(N(CCN2CCC(n3ccc4ccccc34)C2)CC)cc2ccnc(C)c2[nH]1 C1(CC(=O)N(C(C)CC2CC2)C)CN(C(=O)CC2CC(N(C)C)C2)C(C)(C)C1 C1(CNC(COCC(=O)NC)=O)N(C(=O)C(C)Cc2ccco2)CCCC1(C)C N1(C(COc2cccc(C#C)c2)=O)CC(NC(C2CC(F)(F)C2)=O)CC(C)(C)C1 CN1CCN(C)C(C(=O)NCC2CC(NC(c3cnn4c3CCC4)=O)C2(C)C)C1 CCC(C)CC(=O)NCCC(CNC(=O)C(C)(C)c1cnn(C)c1)OC c1(C(C(=O)NC)N(C)Cc2ccc(C(C)(F)F)cc2)cnc(C(F)(F)F)c(F)c1 N1(C(CCOCC(C)C)=O)CCC(CNC(C2(CCF)CCOCC2)=O)C(C)C1 C(=O)(C1CCCn2cnnc21)NCC1C(NC(=O)C2=COCCO2)CC1 CC1(C)CC(C#N)(CNC(=O)COC2CN(C(C3CC34CC4)=O)C2)C1 n1(CC(=O)OCC)nc(C)c(-c2ccnc(C(=O)NC3(COCC)CC3)c2)c1C c1(C(N2CCC(O)C2C(=O)OC)C(=O)NC(CC)C)ccc(OC(F)(F)F)cc1 C(=O)(C1CCc2c[nH]nc21)NCCN(C(=O)CCOc1ccc(F)cc1F)C C1(CNC(CCSCCC)=O)CN(C(C2CC2C(C)C)=O)CC1O C(=O)(CCS(=O)(=O)NC1CC1)NC1C(NC(C(CC)N(CC)CC)=O)CC1 N1(C(CNC(C)=O)=O)CCCCCC1CNC(=O)CN1CCC(C)CC1 N1(C(C2C(COC)C2)=O)CC2(CCN(C(=O)CNC(c3ccc(Cl)cc3)=O)C2)C1 C1(COC)CN(C(c2cc(OC)cc(C3CC3)c2)=O)CCN1C(=O)C(C)C#N Cn1cc(C(N2CCCC2C2(O)CN(C(C3(O)CCC3)=O)C2)=O)c(O)n1 S(=O)(=O)(CCC(=O)N1CCC(c2ncc(-c3ccc(Br)c(C)c3)[nH]2)CC1)NC C(CCC(=O)NCCC1CC(NC(=O)CCc2nnc(C)o2)C1)OCCC c1(C(N2CCC(N(C)C(C3CC3F)=O)C2)=O)oc2ccccc2c1Cl c1(COC)ccc(C(N2CCC(OCCCNC(=O)CC#N)CC2)=O)cc1 C1(NC(C(COC)N(C)C)=O)(CO)CCN(C(=O)Cc2ccnc(O)c2)C1 C(=O)(C(O)CC(F)(F)F)N1CCCC(F)(CNC(c2cncnc2)=O)C1 N1(C(c2cc(C)oc2C)=O)CC2CC(NC(c3coc4ccccc34)=O)C(C2)C1 N1(C(c2cc(OC)n[nH]2)=O)CCC2(CCC2CNC(=O)C=CCN(C)C)CC1 c1(NC(=O)NC2COCCC2(F)F)ncc(F)c(C2CCC2)n1 C12(C(N3CC(C)C(CCNC(c4ccc(C#N)s4)=O)C3)=O)CC(C)(CCO1)C2 c1(CNc2c(C)nn(CC(F)(F)F)c2)cccc2c1CCCC2 c1(CN2CCC(F)(C(N3CC(C(N)=O)NCC3)=O)C2)ccc2c(c1)OC(F)(F)O2 c1(COC)cc(Br)cc(SC2CCC2CO)c1I C1(C(N(CCN(C(c2c(CC)cccc2CC)=O)C)C)=O)CCS(=O)(=O)C(C)C1 C(=O)(CC(CC1CC1)NC(c1cc(OC)no1)=O)NCCOCCC C12(COC(C)(C)C)CN(c3cc([N+](=O)[O-])ccn3)CC1CCO2 N(C(=NCCOC1CCCC1)NCC(=O)Nc1cccc(Cl)c1)C(C=C)C C(=O)(CC(C)P(C)(C)=O)N1CCC(F)(CNC(c2c(CC)n(CC)nc2)=O)C1 N#Cc1ccc(F)c(C(N2CCN(Cc3c(I)ccnc3F)CC2CC#N)=O)c1 c1(-c2cn(C3CCC(C(=O)NC)C3)nn2)cc(Cc2cccc(F)c2)cc(F)c1 C(C)(C)(CC(F)C(=O)N1CCC2(CO)CCCC12)NC(c1c(C)nc(C)o1)=O C(C(O)C(F)(F)F)N(C(C1(NC(C(CSC)OC)=O)CC1)=O)C c1(C2C(C(=O)NCC(CNC(CC=C(C)C)=O)F)C2)c(F)cccc1Br CC(CC(=O)N=c1ccn(C2CN(C(c3nccc4nc[nH]c34)=O)C2)[nH]1)C1CC1 CCCCCCC(C)(CC)C(=O)N(CCCNC(=O)COC1CCOC1)C c1(OC)cc(C(=O)NCCOC2CCN(C(=O)CCC(C)OC)C2)n(C)n1 C1(O)(CNC(C2C(C)=CCS2)=O)CCCN(C(=O)C=Cc2cnn(C)c2C)C1 C1(C(=O)NCC(C)CN(C(=O)COCc2nc(C3CC3)no2)C)COC(=O)O1 Cc1ccc(C(=O)NC(C)(CNC(c2ccnc(S)c2)=O)CC(C)C)c(F)c1 Cc1cc(C(=O)NC2CC(N(C)C(C3CCCC(O)C3)=O)C2)ncc1CO Cc1ccc(Br)cc1C1CCCN1C(=O)C(=O)NC1COC2(CNC2)C1 CC1CC(C(=O)NCCC(F)(F)Cl)CCN1C(C1CC=CCO1)=O C#Cc1ccc(C(=O)NCC2CCC(C(N3CCC(NCC=C)C3)=O)C2)o1 N1(C(c2c(CC)nc[nH]2)=O)CC(C)(C)CC1CNC(=O)Cc1csc(C)n1 CC1CCc2[nH]c(=NC3CC(CC#N)C3)[nH]c(=NCC(C)(O)c3ccco3)c2C1 c1(C(N(CCC(N2C(COC)C=CC2)=O)CCCO)=O)cnccc1NC C(=O)(C(F)C(C)C(F)(F)F)NCCOCCCN(C(C1=C(C)OCC1)=O)C Cc1cc2c[nH]nc2cc1C(N1CC(CCNC(c2cc[nH]n2)=O)C(C)C1)=O c1(C(N2CC(C)CC(C(=O)OC)C2)=O)cnc(C)cc1C.C1CC(=O)N1CCO C(=O)(C(F)(F)C(F)F)NC1C(NC(=O)CCc2cnco2)CC1 CC(C(=O)NCC1CCC1)N(C)C.C1(=O)C(=O)NCCOCCN1C C(CCCC(C)C)(c1n(C(CC)(C)C)nnn1)NC1(C)CCOC1 N1(C(C2CCN(CC)C2)=O)CCC(C2CCN(C(=O)Cc3ccon3)CC2)C1 N1(C(C(CC)O)=O)CCC2(CC1)CC(NC(C1(C)CC1)=O)c1cc(C)ccc1C2 C=CC(CC)CC(=O)NC(CC(F)F)C(=O)N(C1CC(C(N)=O)C1)C C(=O)(C(CC(=O)N1CCN(C(c2ncc(C(F)F)s2)=O)CC1C)C(C)=O)OCC CC1(C)CCN(C(c2ccc(Cl)s2)=O)CC1NC(c1cn(CCCF)nn1)=O C(c1ccc(C(N)=O)cc1)=CC(=O)N(CC(CN(C(C=C(CCC)C)=O)C)O)C c1(OC)ccc(C(N2CC(O)CC2CNC(=O)CCC2(C)CC2(F)F)=O)c(F)c1 C(=O)(CC(CC=C)NC(c1cn(C(C)C)nn1)=O)N1C(C#C)CC1 C(=O)(C1CC(C)Cc2c[nH]nc21)N1CC(NC(COc2cccc(C)c2F)=O)C1 C1(NC(C2C3(CC(NC(c4cc(CC)oc4C)=O)C3)C2)=O)CCCOC1(C)C C1(NC(c2nc(COC)sc2)=O)CCCCCC1NC(c1c(C)cncc1F)=O C1(C(C(=O)N(C(C)CNC(=O)C=C(C)C)CC)C)NC(=O)NC1=O C1(CC(=O)NC2(CC=C)CCN(C(c3cnccc3Cl)=O)C2)CC(=O)NC(=O)C1 C1(NC(=O)CC2CCC3CC23)CC2(C1)CC(C(=O)NCc1ccc(CO)nc1)C2 N1(C(CSCCOC)=O)CC2(C=C(C(=O)Nc3cccc(SC)c3)CO2)C1 Cc1onc(CO)c1C(=O)NC(C)CC1CN(C(c2csc(C)c2N)=O)C1 CC(C)CC(C)(O)CNC(=O)CCN(C)C(C1C2CCCCC12)=O N1(C(c2c(C(C)O)cccc2)=O)CC2(CCN(C(=O)CC(C)C(F)(F)F)CC2)C1 c1(NC(C(=O)NCC2CCCN(C)C2)=O)ccc2c(c1)C(=O)CCO2 C1(NC(C=C(CC)C)=O)CCCCN(C(c2sccc2F)=O)CC1 N1(CC(N2CC(NC(c3c(C(C)C)con3)=O)C(F)C2)=O)CCCCCCC1=O C(=O)(C1CCCc2ncnn21)N1C(CNC(C2CC(OC)C2)=O)CC1 c1(C(=O)NC(CN(C(CCC(=O)NCCC)=O)C)CC)cc(N)ccc1C C1(C(=O)NCCc2ccnc(C)n2)CCOCCN1C(C1C=CCCC1)=O N1(C(C(=O)NC)C)CCC2(CC1)CN(C(=O)C(N1CCNC1=O)C)CC(C)O2 C1(NC(C(C)n2cncn2)=O)CC2C1CCN2C(c1nnc(S)n1C)=O C(=O)(C1Cc2ccc(Cl)cc21)N1C2C(NC(=O)CCc3cnn[nH]3)CC(C2)C1 CC1CC(CC(N2CCOC(CN=[N+]=[N-])C2)=O)CN1C(=O)Cc1cc[nH]c1 C1(CC)CCCN(CC(=O)N(C2CC(NC(C3(CC4CC4)CC3)=O)C2)C)C1 c1(C(=O)NC2CC(N(C(CCC(=O)OC)=O)C)C2)cc(Cl)ccc1F C1(C(C)NC(C2CC(C(=O)O)C2)=O)CN(C(=O)CNC(c2ccco2)=O)CCO1 C1(CC(=O)N(CCCSC)C)CCN(C(c2cncc(O)c2)=O)C1(C)C c1(N(C)CCN2CCOCC2)ccc(S(=O)(=O)NC2(CN(C)C)CCC2)cc1Cl c1(CC)onc(C)c1CNC(c1occc1CNC(c1cc(CO)c(C)o1)=O)=O c1(C(=O)NC(C)(C)CCCNC(=O)C(=O)NC2CC2)ccc2c(c1)OC(F)(F)O2 CCC(CC(=O)N1CCN(C(=O)CCC(C)(C)C#N)CC(C)(C)C1)C(C)(C)C C(=O)(C(CN(C)C)N(C)C)NCC(CC)NC(C1(C(C)C)CC1)=O c1(C(N2CCC(O)(C(C)NC(CSCC#C)=O)CC2)=O)ccc2c(c1)C(C)CN2 N1(C(C2(CC)CC2)=O)CC2(CCCC(CNC(=O)COc3cccc(F)n3)O2)C1 c1(C(N2C(CNC(CN(C)CCO)=O)CC2)=O)cnc(N)cn1 Cc1ccc(C2CC2OCc2cn(CC3C(c4ccccc4)C3(F)F)nn2)cn1 c1(CC(=O)NCC2(NC(COCCCC)=O)CCCC2)c[nH]c2cccc(C)c12 C(=O)(C1=NOC2COCC12)NC(CC)CNC(c1cnc(C(F)(F)F)c(F)c1)=O CN1CCN(C(C2CSC2)=O)CC1C(=O)NCC1CCCOCC1 n1(CC(=O)NCc2cccc(NCC)c2)cc([N+](=O)[O-])ccc1=O c1(C(N)=O)cnc(C(N2CC(Cn3cc(-c4nccs4)nn3)C2)=O)c(Cl)c1 c1(C(N2CCC(OCCNC(c3c(C)onc3CO)=O)C2)=O)cc(F)cc(F)c1 c1(C(=O)NCC2CN(C(C(CC=C)(C)N(C)C)=O)C2)cnc2c(c1)CCOC2 c1(C(=O)NC(COCC)C(=O)NC(CO)C2CCC2)cccc(F)c1 Cc1cccc(C(=O)NC2CC3(C2)CC3NC(=O)Cc2ccno2)c1O C=CCC(C)(CC)C(=O)N1CCCC1CNC(c1cncc(NC)c1)=O N1(Cc2ccc(CCC)cc2)CCOC(C)(CNC(C2CC=C(C)CC2)=O)C1 C1(S(=O)(=O)c2ccccc2)(C(N(C2CCCCC2)CC(=O)OC)=O)CCNC1 c1(C(=O)NC2CCN(C(c3cn(CC)nc3)=O)CC2C)cccc2nc(S)oc12 Cc1sccc1C(=O)NC1CCC(NC(C2CCN2C2CCCC2)=O)C1 C1(CNC(C=C(CC)C)=O)CCN(C(C2(C(=O)OC(C)(C)C)CC2)=O)CC1C N1(C(C(C)=CC(C)(C)C)=O)CCC(OCC(NCP(C)(C)=O)=O)C1 c1(OC)ccc(C(=O)NCc2cnn(C)c2C(=O)NCCC#CCO)nn1 N1(C(c2c(C(C)C)ncs2)=O)CCC2(NC(=O)CN=S(C)(C)=O)CC2C1 CCC(C)CC(C(=O)NCCC1CCOCC1)NC(c1cc(O)cc(F)c1)=O CC(CC(F)(F)F)C(=O)NCC#CCNC(C12CCCC1(C(N)=O)C2)=O C1(NC(=O)Cn2nccn2)CCCN(C(=O)COC2CCC2)CC1F CCC(C(=O)NCC1(CSC)CCN(C(c2ncsc2NC)=O)C1)C(F)(F)F N1(C(C(C)C(C)(C)C)=O)CC2CCC(CNC(=O)C(c3ccccc3)F)C2C1 N1(C(C2N(C(c3c(CC)n[nH]c3)=O)CC2)=O)CC2(CC(N(C)C)C2)C1 N1(C(C=NOC)=O)CCCC(NC(c2cnn(CCOC)c2C)=O)C(F)C1 C=CCC(CCCCC)C(=O)NCC1(NC(c2cc(C)ccc2C)=O)CC1 N#Cc1cc(S(=O)(=O)NC2C3CCCCC23)ccc1NCCc1ccccc1Br c1(OC)ccccc1C(C)=CC(=O)NCC(C)N(C(=O)CCC1CC1C)C C(CCC(O)C(=O)NC1CCC(C(N)=O)C1)NC(c1cc(C)sn1)=O C(=O)(C1c2c[nH]nc2CN1C(c1cc(O)nn1C)=O)NCCCN(CC(C)C)C N1(C(C2(COC(C)C)CC2)=O)CCC(CN(C(=O)CCc2cscn2)C)C1 C1(CNC(C(C)=C(C)C)=O)C(C)CCCN1C(C1CC(C)CC(C)C1)=O C1(C(N(CCn2cncn2)CC)=O)CC(N(C)NC(c2ccsc2)=O)C(O)C1 Cc1nn(C(C)C)c(C)c1C(N1CC(CNC(C2(F)CC2C)=O)C(C)(C)C1)=O C1(C(=O)NCc2n(CCC)ccn2)CCN(C(=O)c2ccsc2C)O1 c1(C(N(CCN(C(=O)C(N)=O)C)C)=O)ccc(C(=O)OC(C)(C)C)cn1 c1(C(N2C(CCCNC(C=CCC)=O)CCC2)=O)cnc(O)n(C)c1=O C(=O)(CCCCCC)N1CCC(C(C(=O)N(CCCCCC=C)C)C)C1 C1(C(=O)NCC(C(=O)N(CC(O)CF)C)O)CC(=O)NC(=O)C1 C1(CNc2cc(Oc3c(OC)cccc3)ncn2)CN(C)CCC1(F)F C1(C(N2CCCCC(CNC(c3c(C)nc(C)[nH]3)=O)C2)=O)CCc2ncsc2C1 c1(C(=O)NC(C)CC(C)NC(=O)C(C)Cc2cnn(C)c2)cnc2ccccn12 c1(C(=O)NC2CCC(C(=O)Nc3cncc(F)c3)CC2)n[nH]c2c1CS(=O)(=O)C2 C12(C(N(CCNC(c3cc(C)c(C)s3)=O)C3CC3)=O)CCCN(CC1)C2 Cc1cc2c(cc1C)OC(C(=O)NC1CCN(C(c3ccco3)=O)CC1C)C2 C1(C(=O)NCCN(C(=O)C(O)C(C)C)CCOC)C(C)OC(C)C1C C(=O)(C(F)(F)C(O)CC)NC(CC=C)CNC(c1cccnc1O)=O c1(C(N(C)CC2CCN(C(c3c(C)nc(C)[nH]3)=O)C2)=O)cccc(N)c1Br c1(NC(=O)COC(c2cnc(CCC(F)(F)F)s2)=O)nccc2ccccc12 c1(OC)ncc(NC(C2CCCN(C)C2)=O)cn1.C1(=O)CO1 S(=O)(=O)(c1c[nH]c(C(N2CCN(C(=O)CCCC(N)=O)CC(O)C2)=O)c1)N(C)C C1(n2cc(CCN(CC)CC)nn2)CN(C(=O)NC2CCOCC2)CC1C N(S(=O)(=O)N(C)C)CC(=O)NC1(COC)CN(C(=O)CC(C)(C)C)C1 Cc1cc2nc(NCC3C4CN(C(=O)CCC5CCC5)CC34)cc(=O)n2o1 c1(C(C)C)ccccc1C(N1CCOC(CN(C)C(C23CSCC2C3)=O)C1)=O N1(C(C)=O)CS(=O)(=O)CC1C(=O)NCC(O)CNC(=O)CCF c1(COCC(=O)NC2C(CNC(C(C)(C)OCC)=O)C2)ccc(CC#N)cc1N CC(C)C(F)C(=O)N1CC(CNC(C2CS(=O)C2)=O)C(O)C1 c1(OC)cccc(N2CCC(NC(=O)Cc3ccccn3)C2)c1-c1nn[nH]n1 c1(C(N2C(CCNC(C3(c4ccn(C)n4)CC3)=O)CCC2)=O)cccn(C)c1=O C1(CN(C2CCCCC2)C(c2c(Br)nc(C)s2)=O)CCCCS1(=O)=O C12CC3(COC1C3)NC(c1nnnn1C)CCCN2.C1(CN(C)C)CC2CC2C1 c1(C(=O)NC(C)CCCNC(c2cc(CO)[nH]n2)=O)c2ccccc2nn1C C(CCC(=O)N(C1CC(NC(=O)C(C2CC2)N(C)C)C1)C)=CC(C)C CON(C)C(=O)C(CNC(C1CC(O)CN1C)=O)C(C)(C)C C(=O)(C(O)P(C)(C)=O)N1CCCC(CCNC(c2cc(COC)on2)=O)C1 N1(C(CN(CCCCCC)C)=O)CCC(COC)(NC(=O)C(C)(C)SC)C1 C1(C2CCCOC2)(NC(=O)CC2(C3CC3)CC2)CC1 C1(NC(CC2(OC)CCC2)=O)CC2CN(C(=O)CSC(F)F)CCN2C1=O c1(C(C(=O)N(CCN(CC)CC)C)NC(=O)CCn2cnnn2)cn(C)nn1 N1(C(C2C(CC)C2)=O)CC(NC(=O)C(C)CC(N)=O)CCC1C N#CC1CCC(C(=O)NCCNC(C2CCSCC2)=O)C1 c1(C(=O)NCCn2cc(C(=O)NC(CCOC)C)nc2)cnccc1C Cc1cc(Cl)ncc1CC(N1CC(O)(CCNC(=O)CCSC(F)(F)F)C1)=O C(C(C)CC(C)C)NC(c1n(CC=C)nnn1)CCC1CCCC1 C(=O)(CCCCCCn1cc(C2CCOCC2O)nn1)NCC(C(C)(C)C)O N1(N(CC=O)CCOC)CCC(O)C(O)C1.c1(C=O)cn(C(C)C)nn1 c1(C(=O)NC(C)C(C2CCCCC2)NC(=O)C=CBr)ccnc2[nH]nnc12 C(=O)(C1=C(F)CN(C(=O)CC(C)OC)CC1)NCC1(OC)CCCC1 Cc1nccc(=NC(C)C2CCCN(C(=O)CC(C)n3ccnc3)C2)[nH]1 C1(CNC(c2n[nH]cc2[N+](=O)[O-])=O)CN(C(C2(O)COC2)=O)CCC12CCC2 O=[N+]([O-])c1cccc(N(S(=O)C2CNC2)CC2CC2)c1 C(=O)(C(CC(C)(C)C)N1CCCC(C(F)F)C1)NC(CC)C C1(CN(C)C(C2CC(O)C2)=O)CC(F)CN1C(C1CCCCO1)=O CCC(C)(C)C(C)NC(c1coc(CNC(=O)CN(C(=O)C(C)C)C)n1)=O c1(C(N2CCC(C(C)NC(c3c(C)cn(C)c3)=O)C2)=O)cc(Cl)ccc1C(C)C C1(CNC(C2CC23CCOC3)=O)CC(N=c2[nH]c(Cl)nc3[nH]cnc23)C1 C(=O)(CC(C)(C)C(F)F)N1C(C)(CNC(C2(C)CNC(=O)C2)=O)CCC1 N1(C(CC(CNC(c2ccc3[nH]ccc3c2)=O)OC)=O)CC2C3CCC(C3)C2C1 N(C1c2ccccc2CC1NC(C1CCS1(=O)=O)=O)C(CN(C)C)=O n1(CC)cnc2c(NC(c3csnn3)C)[nH]c(=NCC3CCC4CC34)nc12 CC1(C)CC=C(C(=O)N2CCC3(CC3NC(=O)CC3CCOC3)C2)CC1 CCCN=c1[nH]c(N(C)Cc2ccc(C(C)(C)C)nc2)nc2c1CC(C)CC2 Cc1noc(C2CCC2ONC(n2nnc(-c3ccccc3)n2)=O)n1 Cc1nn[nH]c1CC(=O)NCC(=C1CN(C(=O)CCc2cn(C)cn2)C1)F C1(C(C)C)CN(C(=O)COc2cnn(C)c2)CCC1NC(c1cocn1)=O N1(C(C(N2CC3CC3C2)C)=O)CCc2sc(C(=O)NC3CN4CCC3CC4)cc2C1 N1(c2ncc(C)cn2)CCC(NC(=O)C(F)(F)C2(O)CCC2)C(CO)CC1 c1(C(=O)NC2C(=O)NOC2)cccnc1-c1ccc(C2(NCCO)CCC2)cc1 C1(C(=O)NC(C2CS(=O)(=O)C2)C)CCc2nn(C)c(C(F)(F)F)c2C1 c1(C(N2C(CNC(CC3CC(=C)C3)=O)CC2)=O)cc(S(N)(=O)=O)oc1C C1(O)(C(C(=O)OCC)(F)F)CCN(C(=O)NC(C2CCCC2)C)C1 C1(NC(C(C=C)(C)O)=O)(COC)CCN(C(=O)COc2ccsn2)CC1 C1(C2CCCN(C(C34CCCC(C3)OC4)=O)C2)(NC(=O)Cn2cccn2)CC1 C1(C(=O)NC2CN(C(c3ncoc3-c3ccc(F)cc3)=O)C2)COC2(CCC2)C1 c1(CC)cccc(C(N2CC(O)(CNC(C3CC(C4CC4)=NO3)=O)C2)=O)c1O N1(C(=O)C=Cc2ccco2)CC(O)C(O)C12CCC2 N1(C(CCC(C)OC)=O)CCC=C(CNC(c2ccc(C)nc2C)=O)C1 C1(NC(c2nc(NC(C)=O)sc2)=O)CS(=O)(=O)CC1NC(=O)COC(F)F C(C)(C)(C(=O)N(C(C)C(=O)N(C1CCC1C)C)C1CC1)SC N1(C(c2cn(CC=C)nc2)=O)Cc2n[nH]cc2C1C(=O)N(C)CC1CC(=C)C1 C12(NC(C3N(C(C)=O)CCC3)=O)COC(C1)C(NC(=O)CSCC(C)C)C2 Cc1coc(C)c1C(N1CCC(CNC(=O)CC2CC2c2ccccc2)C1)=O N1(C(c2scc(C)c2)=O)CC2CCC2(CC(=O)NC2CC23CCCC3)C1 C(=O)(C1=Cc2ccccc2OC1C(F)F)NCc1cn(CCCC(=O)O)nn1 [N-]=[N+]=Nc1cncc(CNC(c2ccccc2-n2cc(Br)cn2)=O)c1 N1(C(c2c(CC)nc(C)[nH]2)=O)CC(NC(=O)C(c2cccc(O)c2)C)C2(CC2)C1 Cc1ccc(N2CCC(CNC(CC(C)C)c3cn(CCCO)nn3)C2=O)cc1 CC(CNC(N1CCCC1c1cncn1C)=O)CC(F)F N1(C(C)C)C(=O)CN(C(C2(N(C)C(=O)C3CC3)CC2)=O)CC1(C)C N1(C(CCSc2nc(C)sc2)=O)C2CCC1CC(CNC(C13CC(CO1)C3)=O)C2 c1(COC)csc(CN2CCCC2C(c2ccccc2)C(=O)NCO)n1 n1(Cc2ccn(C)n2)cc(C#CCNC(=O)C(C2CC2)C2CC2)nn1 N1(C(C2CCC(CN(C)C)O2)=O)CCc2ccccc2C(NC(=O)C=CCF)C1 C1(OCC(N2CC(O)(COC)C2)=O)CCCN(C(=O)C(C)C(=O)OC(C)(C)C)C1 C(=O)(CCN=c1[nH]c(C)cc(=NC(C)c2n[nH]c3c2CCCC3)[nH]1)NC C1(NC(C=C(CC)CC)=O)C2CC(O)C1N(C(=O)C1=COCCO1)C2 CCCC(C)C(=O)N1CCC(CN(C(=O)Cc2cc[nH]c2)CC)CC1 N1(C(c2[nH]cc(C)c2)=O)CCN(C(c2cn(C)cc2C)=O)C2CCCCC2C1 CC(C)(C(=O)N1CCC(C2(C)N=N2)C1)C1=CCN(C(C2CCC(=O)N2)=O)C1 C1(C)(C(=O)NCC(CC)NC(c2cc(C(C)C)no2)=O)CCCOC1 C1(N(C(=O)C(Cc2ccoc2)N(C)C2CC2)CCCC)CCN(CCO)CC1 C(CO)(C(=O)NC(C(N)=O)C1CC1)NC(CN(C)C1CC1)=O N1(C(CSC)=O)CC(NC(c2cc(C(C)(C)C)no2)=O)C2CC2C1 C1(CC(N2CC(OCCNC(CCc3c(C)ncs3)=O)C2)=O)CCCCN1C C(=O)(C(C(=O)N1CCC(CNC(=O)CC=NO)C1(C)C)C(C)C)OCC c1(C(=O)NC2C(CC)CN(C(c3ccc(F)s3)=O)CC2)cc(OC)c(O)c(N)c1 c1(OC)c(C(N2CCC(CNC(C3COC(=O)C3)=O)CC2)=O)occc1=O C(=O)(C1=CC2CCCC12)NCC1CC(NC(c2ncc(C)nc2)=O)C1 c1(C(=O)NCCC23COC(CO)(C2)C3)cccc2c1CCS2(=O)=O c1(NC2C(C)CN(C(=O)Cn3cnnn3)CC2C)nc2cccc(F)c2s1 C1(CNC(C2CN(C(C)=O)C2)=O)CCCC2(CN(C(=O)CCCCC#N)C2)O1 C(=O)(C(O)C(F)(F)F)N1C(C(C)NC(Cc2c(C)cnn2C)=O)CCC1 N1(C(C(c2cn(CC)nc2)=O)=O)CC(C)CN(C(C2CS(=O)(=O)C2)=O)CC1C c1(C(N(C(C)C(=O)NC(CCC#N)c2ccccc2)CCO)=O)cc(O)nc(O)c1 N1(C(C(C(CC)C)O)=O)CCC2(CC1)CCN(C(=O)CCOC(C)C)C2 C1(NC(CC2(N(C)C)CC2)=O)COCCC1NC(C1CCCN(S(C)(=O)=O)C1)=O N1(C(COC(C)C)=O)CC2CC(NC(=O)C(C)N(C)C)C2C1 c1(OC)ccc(C(=O)NCC2CN(C(=O)C(CC(C)C)N(C)C)CCO2)c(O)c1 C1(CC(N2C3CC(NC(c4c(C)ccs4)=O)(C3)C2)=O)CC2CC1C1CC21 Cc1cc(-c2c[nH]c(=NCc3c[nH]nc3C(F)(F)F)s2)ccc1CN(C)C CC1=CCC(C(N2CCCC2(C)CNC(=O)CC2CC(=O)NC2=O)=O)CC1 N1(C(CC(C)C)=O)CC(NC(c2ccc(F)c(Cl)c2)=O)CC2(CCC2)C1 c1(C(=O)NCC(C)NC(=O)CN2CCOC2=O)cc(S(N)(=O)=O)oc1Cl c1(C(=O)NCC2N(C(COCC(C)C)=O)CCC2)ccc(OC2CCC2)cc1 N1(C(COCCC(C)C)=O)CCC(C)(CNC(=O)C(C2CCC(F)(F)C2)O)CC1 CCC(O)CC(=O)NC1(C(=O)N(C)CC2COCCO2)CC1(C)C c1(CC)c(C)nn2c(C)cc(C(=O)NC(CO)C3(C)CC3)nc12 c1(C(N2CCN(C(C3=CC(C)CC3)=O)CC2CO)=O)nn(C)c2c1CCC2 CCCC(O)CC(=O)N1CCC(C)(NC(C2CCCCC2n2cccn2)=O)C1 c1(C(=O)NC2CC(NC(C3CC4C=CC3C4)=O)C2)cn2c(n1)CCC2 CCC(CCCC(=O)NCCCF)NC(c1cnnn1C1CC1)=O NS(=O)(=O)c1sc(-c2ccccc2)nc1C(=O)N(C1CC1)CC1CCOCC1 C1(n2cc(C(=O)OC)nn2)CN(N2CCC(N3CCCCC3=O)CC2)CC1O C1(CC(=O)NC(COC)CNC(=O)CC2CC=CCN2C)CCCNC(=O)C1 c1(OC)cc(C(=O)NCC#CCNC(=O)C(C)C(C)(F)F)cc2c1OCCO2 C1(CC(C)NC(=O)C=Cc2cscn2)CCN(C(c2c[nH]ccc2=N)=O)CC1 C1(C(N2C(CO)CC(NC(c3cc(Cl)c[nH]3)=O)C2)=O)CCc2ccnn2C1 C1(NC(c2cncc(OC)n2)=O)CN(C(c2ccccn2)=O)CC1C1CC1 C(C(C)C(=O)N1CCCC1C(=O)NCC(CO)N(C)C)SC CC1OC2(C)CC1(C(=O)NC13CC(NC(=O)C4=CCCCO4)(C1)C3)C2 N1(C(CC2(N(C(C3N(C(C)C)CCC3)=O)C)CC2)=O)CCOC2CCC12 Cc1cccc(-n2cc(C3(C)CCCO3)nn2)c1 N1(C(C2(C#N)CCOCC2)=O)CCC2(CCCCC2NC(=O)C=CCF)CC1 C(CC(C(C)(C)C)NC(C1(C2CCCCO2)CC1)=O)N(C(=O)CNC(N)=O)C C1(CC(=O)NCCCN(C(C2CCCCO2)=O)CC)COCCN1C1CCCC1 c1(CC(=O)NC2CN(C(=O)Cc3ocnc3C3CC3)C2)csc(-c2cccs2)n1 c1(CC)ccc(C(C)C(=O)N(C)CC2CCCN2C(C2(CC)CC2)=O)cc1 N1(C(CCOCC)=O)CC(NC(=O)CC(c2ccccc2F)NC(N)=O)C(C)C1 Cc1cc(C(=O)NCC2(C(=O)NC34CCC(C3)OC4C)CCCC2)ncc1F C1(NC(C(C2(C)CC2)NC(c2c(C)cccc2)=O)=O)CC2(CCC2)C1O c1(C(=O)NC2(C3N(C(C(CC)SC)=O)CCC3)CC2)cccc(Br)c1F c1(C(=O)OC(=O)C(c2c(C)nn(C)c2C)C(=O)NC)cc(C(=O)OC)cc(Br)c1 c1(OC)ccc(C)cc1C(=O)N(C1CCCN(C(=O)Cc2ccc(C)nc2)C1)C C1(NC(C2CCC(=O)O2)=O)COCCN(C(=O)Cc2cscn2)C1 c1(OC)ccc(CC2CCN(CCC=CC(C)(C)N)C2)cc1 C1(N(C(=O)Cc2ccc(C)s2)CC)CCN(C(c2ccc(C(N)=O)o2)=O)CC1 C(=O)(N=S(C)(=O)CCCCN)c1cccc(CCC#N)c1 N1(C(c2c(C)nn(CCO)c2)=O)CC(CNC(=O)CC2C=CCCC2)CC(C)C1 c1(COC)nc(C)c(C(N2CCCC(CCNC(=O)Cc3ccsc3)C2)C)o1 N1(C(C(CC)CC)=O)CCCC(O)(CNC(C2CCC2Cc2ccccc2)=O)C1 C1(NC(c2csc(N3CCCCC3)n2)=O)CCCCCN(C(=O)CCCF)C1 c1(OCC)cccc(CC(=O)N(C)CCN(C)C(C2CC=CCO2)=O)n1 C1(CNC(c2cc(C)oc2)=O)C2CCC(C2)N1C(=O)CC1CCCO1 N1(C(CC=C)=O)CC2CC(C(=O)NCCc3c[nH]nc3C)CC2C1 CC1(C)CCCC(C(=O)NCCC2(CNC(=O)CSS(C)(=O)=O)CC2)CC1 C1(CC=C)(C(=O)NC2CCN(C(=O)CCCc3ncc(C)o3)C2)CCCCC1 C1(CSC)(CNC(=NC)NCCCNC(C2CCC2)=O)CCCCC1 N(C(=NCCNCC(C)(C)O)NCc1cccc2c1OCC2)C1C(C)C1 N1(C(C(CCC)c2ccc(Cl)cc2)=O)CCN(C(=O)C2=CCOC2)CC1C c1(C(=O)NCC(CC)NC(c2cnn(CCO)c2N)=O)c(C)noc1C(F)F N1(C(c2cc(C3CCC3)[nH]n2)=O)CCC2CCN(C(=O)C(F)=C3CCC3)CC2C1 Cc1cn2cc(C(=O)N(C(CNC(=O)CCCn3ccnc3)C3CC3)C)nc2s1 S1(=O)(=O)c2cccnc2NC2COCCN12.C(C(O)C1CCC1)N(C)CCO CCCCC(CNC(c1sccc1NS(C)(=O)=O)=O)NC(=O)C(C)C(C)O C1(CC(=O)NC2C(NC(c3c(C(=O)OC)cco3)=O)COC2)CN2CCC1CC2 C(N(C)N1CCC(C)(N2CCCC2)CC1)c1cccc(C)n1 C1(N(C(c2cnc(C(C)C)[nH]2)=O)C)CCN(C(C2(F)CC=CCC2)=O)CC1 C1(SC)COCC1NC(=O)C(Cc1cn[nH]c1)NC(=O)CCn1cnc(=N)[nH]1 N1(C(CN2C(=O)CC(C)(C)O2)=O)CCC2(CC1)CC(NC(C1CSCCS1)=O)C2 C(CCC(=O)NC(C)CC(C)NC(=O)CNc1ccccn1)N(C(C)C)C CC(F)(F)CCCC(=O)N1CC2CCCC1(CNC(C1(O)CCCCC1)=O)C2 c1(C(N2CCC(c3ccc(OC)cc3)(O)C2)=O)c(Cl)nc2sccn12 c1(C(=O)NCC23C(CN(C(C(C)(C)N(C)C)=O)C2)C3)ccc(N)c(F)c1F C(=O)(C1CCc2ccc(C)cc21)NC1CCN(C(c2nn(CC)nc2C)=O)CC1 N1(C(=O)Nc2ccc(C(F)(F)F)c(-c3ccno3)c2)CCCC2COCC12 C1(C(=O)NCC(CNC(c2nnn(C)c2N)=O)(C)C)CCCCS1(=O)=O CN1CCCCC1CC(=O)NC1CCC(N(C)C(C2COC(=O)N2)=O)CC1 N1(C(CNC(=O)OC)=O)CCCC2CN(C(c3ccn(CCF)n3)=O)CC12 C(C)(CC(=O)NC(C)CC(=O)NCC1(C(C)C)CCCC1)=C(C)C C(=O)(C#CC1CCOCC1)N1CC(C2CN(Cc3oc(C)c(CO)c3)C2)OCC1 C(=O)(C(C(C)CC1CC1)N1CCCC1c1ccc(SC)cc1)NCC c1(C(=O)NC2CCN(Cc3c(C)ccc(O)c3)CC2)ccc2c(c1)OC(F)(F)O2 C1(C(=O)NCC(=C)CCNC(c2coc(CC)n2)=O)CCn2c(Br)cnc2C1 C(=O)(CC(CN(C)C)C(F)(F)F)NCC1N(C(c2c(C(C)C)[nH]cc2)=O)CC=C1 c1(C(=O)NCC2(NC(Cc3c(C)non3)=O)CCOCC2)cccc([N+](=O)[O-])c1 c1(C(=O)NCCC2CCCN(C(=O)Cn3cccn3)C2)nnc2ccccn12 N1(c2cc(OC)nc(COC)n2)CCN(C(=O)CSC(F)(F)F)CC(O)C1 c1(C2CCC(=O)NC2=O)nc(=NC2CN(C(C3CC4CCC3O4)=O)C2)cc[nH]1 CC(CN(C)C)CCC(=O)NCC(C)CNC(=O)CCCc1cccc(Cl)c1 C1(NC(CCNC(Cn2ccc(C)n2)=O)=O)CCSC(C)C1 c1(OC(CC)C(=O)NCCC2(CNC(C3CNC(=O)N3)=O)CC2)ccccc1F c1(C(=O)NCC2OCCN(C(C(C)SC(C)C)=O)C2)cc(Cl)nnc1O NC1CCC2(c3nc(-c4ccccc4)nn3C3CCCCC3)CCC12 N1(C(C2(COC(C)C)CC2)=O)CCOCC(C(=O)N(C)CC2CCCC3CC23)C1 C(C(C)CC(=O)NCC1CN(C(=O)C(C)(F)F)CC1c1cncn1C)OC Cc1cc(CC(=O)NCC(CO)NC(=O)C(C)(C)c2ccccc2)n[nH]1 c1(OC)ccc(C(N2CC(CNC(C3COC(C)(C)CO3)=O)C(C)C2)=O)cc1F c1(C(=O)NCC(CNC(C(CC(C)C)F)=O)(C)O)cc(Cl)c2n[nH]cc2c1 c1(OC)cnc(SC)nc1N(C1(CO)CNC1)C(c1ccc(Br)cc1)=O C1(NC(CC(CC)(C)C)=O)CCN(C(c2cccc(C(C)=O)c2)=O)CCC1CO c1(C(N(C)CC2CCN(C(C3(OC)CCCC3)=O)C2)=O)cc2sc(C)cc2s1 N1(C(C(C=CC)O)=O)CCCC(CCNC(=O)Cn2ncccc2=O)C1 c1(C(C)C)ccc(CC(=O)NCCNC(C2CC(C)OC2=O)=O)cc1F Cc1nc(-c2cccc(C3CC3C(N3CCCC(F)C3)=O)c2)c2ccccc2n1 c1(OC)c(C(=O)NCCN(C(=O)CC2COCC(C)(C)O2)C)ccnc1Cl C#CCCC(O)C(=O)NCC(CO)NC(=O)Cn1cc(Br)c(=N)[nH]1 N1(C(=O)NCC(COC)F)CCC(C(C)(C)F)C1 c1(C(N(CC(C)N(C(CC=C=C)=O)C)C)=O)c(C)coc1C(C)(C)C c1(C(=O)NC2CN(C(CS(CC)=O)=O)CC23CC3)cccc2c1OCC2 C(=O)(CC1OCc2ccccc21)N1CCC(NC(C=C(C)C)=O)C(O)C1 N1(C(CSC)=O)CCN(C(C2(c3ccc(Cl)c(Cl)c3)CCC2)=O)CC1C C1(NC(C)=O)CCN(C(=O)N(S(C)(=O)=O)C)C(C)C1 C(Cc1ccco1)(C(=O)N(C)Cc1ccns1)NC(CNC(CCC)=O)=O c1(C(=O)NCC2(O)CCCN(S(=O)(=O)CCCCCl)C2)cccc2ccnn12 C1(C(=O)NCCC(CCC)O)CCN(C(=O)CC2CC=CC2)C12CCC2 CCCC(C(=O)N(C1CN(C(=O)CC(C)C2CC2)C1)C)NC(=O)OC(C)(C)C N1(C(c2ccc(OC)nn2)=O)CCN(C(C2CCC(=O)N(C3CC3)C2)=O)C(C)C1 C1(C(=O)NC(C2CN(c3cc(F)ncn3)CCO2)C)CCc2nn[nH]c2C1 C1(C(N(C)Cc2cnc[nH]2)=O)CCC(O)CN1C(C1CCCC(=O)C1)=O CC(CC(=O)N1CCN(C(c2cc3ccsc3[nH]2)=O)CC12CCC2)CC(C)(C)C c1(C(=O)NC(C2(CNC(C3COC(=O)C3)=O)CC2)C)ccc(CO)o1 C1(NC(CCC(C)(C)C)=O)CN(C(=O)CN2C(=O)CCC2=O)CC(C)(C)C1 S(=O)(=O)(c1ccccc1)NCC(=O)N(CC(O)CNC(C1(F)CC1)=O)C C1(OCC)CC(C(=O)NC(C)C(C)NC(=O)C(C)OCC(C)C)C1 c1(OCC)ccccc1C(N1CCCC(C2CCCCO2)C1)C(=O)NC(C)CC CC1C(C(=O)N(C)CCN(C(=O)CCc2ccc(C(F)F)cc2)C)CCN1C C1(C(C)NC(=O)CNc2ccccc2-c2ccccc2)CCC(F)(F)CO1 N1(C(CC(=O)OC)=O)CCCC(F)(C(=O)NCC2(OC)CC2)C1 c1(C(C)C)nn(C)cc1C(=O)NCC1C2CN(C(C3CCOC(C)C3)=O)CC12 c1(NC(C2C(NC(c3scc(C)n3)=O)CCCC2)=O)ccc(C)c(C#N)c1 C(=O)(C1=CS(=O)CCC1)NC(C(C)C)CNC(C1CC(n2cnnc2)C1)=O N1(C(CC2CCN(C(=O)NC3C=C(C)CS3)C2)=O)CC2(CCN2C)C1 CC1(C)OC2(CNC(C3CCS3(=O)=O)=O)CC1(NC(C1CSCCS1)=O)C2 c1(C(=O)OC)cc([N+](=O)[O-])cc(Cl)c1N(C)CCN(C(=O)C=CC1CCOC1)C Cc1c(-c2cn(-c3ccc(Cl)c(-c4nn[nH]n4)c3)nn2)cccc1Br N1(C(COC)=O)CCCCC(NC(=O)CS(=O)C(F)(F)F)CC1 N1(C(C2CCN(c3ccn(C)n3)C2)=O)CCN(C(=O)C(C)(C)C#N)CC1CCO CC1COC(c2ccccc2)CN1C(=O)Nc1nc(CN2CCOCC2)no1 c1(C(=O)NCCCN(C(CCn2c(C)cc(C)n2)=O)CCO)ccc(C)c(F)c1 C1(NC(c2c(CNC(c3ncn(C(C)C)c3)=O)n[nH]c2)=O)CC(CO)CC1O CC1CCN(C(c2cnc(Cl)cc2Cl)=O)CC1CNC(=O)C(c1cnn(C)c1)=O N(C(=NC)N1CC2C(C(F)F)C2C1)C1CC(c2c(OC)cccc2)C1 c1(COC)cnc(CC(=O)NC(C)CN(C(=O)COC2CCCCC2)C)[nH]1 N#CCCCC(=O)NCC1CCCC1NC(c1cnc(C2CC2)o1)=O Cn1cnnc1CCCC(=O)NC1CCC1NC(c1ncoc1-c1ccco1)=O C#Cc1ccccc1CC(=O)NC(CNC(=O)COc1cc(Cl)ccc1Cl)CC C1(CNC(c2sc(C)c(O)n2)=O)CCC(C)CN1C(c1cnn2c1OCC2)=O C1(C(N2C(CNC(c3cn(CC(F)F)cn3)=O)CCC2)=O)CCc2nnnn2C1 n1(CC(=O)NC2CCN(C(C3N(CC)CC3)=O)C2(C)C)ccc2ccccc12 c1(C(NOC)=O)ccc2ccc(NC(c3c(Cl)cnn3C)=O)nc2c1 C1(CN(C(C(C)OCC(C)C)=O)C)CCN(C(c2ccc(OCF)cc2)=O)CC1 CN1CCN(C(C2CCCN(C(=O)CC3CCC(C)(C)O3)CC2)=O)CC(O)C1 N1(CCCNC(c2cc([N+](=O)[O-])c[nH]2)=O)CCCN(Cc2ccccc2)CC1 c1(COC)nc(NCCCNCc2cccs2)cc(=NCc2csc(C)c2)[nH]1 Cc1c(F)ccc(C(=O)N(C)CCN(C(C2CN(C)CC(C)O2)=O)C(C)C)c1N N1(C(C2CN(C)C(=O)N2)=O)CCC2(CC1)CCN(C(C1CCCOC1)=O)CC2 C1(CN(c2nccnc2C#N)C)CN(C(=O)CN(C)S(=O)(=O)N(C)C)CC12CC2 c1(NC(C(=O)NC2C(CNC(C(CC3CCCC3)OC)=O)C2)=O)cc(C)ccc1Cl c1(OCC(=O)NCCC(CNC(=O)C=Cc2cccnc2)O)ccc(F)c(Cl)c1 N1(C(C(CC=C)C)=O)CCC2(CC1)OC1(CO)CC2(NC(C2CC(F)(F)C2)=O)C1 N1(C(c2ccc(CO)cc2)=O)CCC2CCN(c3ncc4ccsc4n3)CC2C1 C1(NC(C2C(NC(C(CC)(C)CC)=O)CCO2)=O)CCOC2(CCC2)C1 N1(C(Cn2nnc(C)n2)=O)CC2(CCCCN2C(c2cc(Cl)cn2C)=O)C1 c1(C(N(CCCNC(Cc2cn(CC)nc2)=O)CC)=O)cc(C(F)(F)F)ncn1 c1(C(=O)NC2CC(N(C(CCCc3cc(C)no3)=O)C)C2)c(C)ccc(Cl)c1O c12cccn1CC(=O)N2.C1(N(C(N(C)C)=O)C)CC1(C)C N1(C(C2(CC=C)CC=CC2)=O)CC2ON=C(CNC(c3cnc(CC)s3)=O)C2C1 C1(C(N(C2CCCN(C(COCCOC)=O)C2)CCO)=O)OCCN(C)C1=O Cc1cc(CN=C(NC2CC2)NC2CC3CCCCN3C2)ccc1[N+](=O)[O-] C=C(CNC(c1cc(F)ccn1)c1nnnn1CCC(=O)OCC)C(F)(F)F c1(C(=O)NCC2(CN(C(C3C(C=C)C3)=O)C)CC2)cnc(O)c(Cl)c1 C1(C(=O)NC2CC2NC(C2(C)CCOCC2)=O)(OCC)CCSCC1 CC1CCC(F)(F)CN1C(=O)C(C)(C)CN(C(=O)CCc1cnccn1)C N1(C(c2cc(CNC(CCc3n(C)cnc3)=O)on2)=O)C2CCC1CC(CO)C2 Cc1nccc(N(C2CCCN(C(=O)CCC3CCC(C)O3)C2)C)n1 C1(NC(CC2CCCN(C(CC3CC(N(C)C)C3)=O)C2)=O)CCNC(=O)CC1 Nc1ccc(Br)cc1C(=O)NC1(CCNC(c2cnn(CCCF)c2)=O)CC1 c1(C(=O)NCC(N(C)C(C23CC4CC2C3C4)=O)C2CC2)cc(F)cnc1O C1(C(=O)NC23CC(NC(c4c(C)nccc4)=O)C(OC2)C3)CNC(=O)C(C)(C)C1 C(CCCCC(=O)NCC1(F)CN(C(=O)C(F)C2CCOC2)C1)OCC c1(C(N2C(C)CC(NC(C3(COCC)CC3)=O)C2)=O)cc(C)c(F)cn1 CCC(C(=O)NC(C(=O)OC)C1CC1)N(C)C(C1COC(=O)N1)=O c1(C(=O)NC2C(C)CN(C(CC(CC)CC)=O)CC2C)sc(S(N)(=O)=O)cc1C Cc1ccc(=O)n(CC(=O)NCC(C)(C)NC(c2conc2C2CCCO2)=O)c1 N1(C(CNC(=O)NC)=O)CCC(NC(c2cncc(C)c2Cl)=O)CC1C1CC1 C#CC1(C(=O)NC2CCC(C(=O)NCC3(Cl)CC3(F)F)C2)CCCCC1 CC1CCCCCC1(c1nnnn1Cc1ccco1)NCC12CC(F)(C1)C2 CC1CC(=O)NCCN1C(c1cc(CN(C)C)[nH]n1)C(=O)Nc1ccc(F)cc1 C(CCCCCCCO)=CC(=O)NCCN1C(=O)CC(NC(CC(CC)C)=O)C1 c1(NC(C)=O)ncc(S(=O)(=O)N2CCN(Cc3c(O)cccc3O)C(C)C2)s1 C1(NC(C(=O)NCC2(F)CC(CN)C2)=O)C2Cc3ccc(Br)cc3C12 N1(CCC)CCC(CNCCc2cc(OCC)n[nH]2)CC1 c1(NC(C(Cc2ccoc2)NC(=O)CCn2cnnn2)=O)cccc2[nH]ccc12 C(=O)(C(O)CCS(C)=O)NCCCN(C(=O)CCCNC(=O)C1CC1)CC CN1CCC(C(=O)NCC2(NC(c3cc(CN(C)C)c[nH]3)=O)CCOC2)CC1=O c1(C(N2CCC(CCn3cc(-c4cncc(F)c4)nn3)CC2)=O)cncc(Cl)n1 N1(C(CCCCC(C)C)=O)CC(C)OC2(CCN(C(C3CC=CCC3)=O)CC2)C1 N1(C(COCCOCC#C)=O)CC(C2(NC(=O)C=CC3CCOCC3)CC2)C1 C1(C(=O)NC(CC)CC(C)C)CCOCCC1NC(=O)OC(C)(C)C C(CC(=O)N1CCOCC1CCO)(C(F)F)NC(CCC(=C)Cl)=O CCC1=C(C(=O)N2CCOCC2C(N2CCOCC(O)C2)=O)CCCO1 C(c1cncc(O)c1)=CC(=O)N(C)CC1CC(F)CN1C(c1ccccc1F)=O C(CCCC(=O)N1CC(NC(c2nc(C(C)(F)F)cs2)=O)CC1C)NC(C)=O C(=O)(C1=NOC(CNC(c2ccc(CF)cc2)=O)C1)N1C(C)(CC)CC1 c1(C(N2CC(OC)C(NC(c3cc(C)cs3)=O)C2)=O)csc2c1C(C)(C)CCC2 C1(C(=O)NC(C(N)=O)CO)C2CC3C(C2NC(c2ccccc2F)=O)C13 C(=O)(C(CN(C)C)C(C)C)NCC1C(CC)CCN1C(=O)Cc1cnccc1Cl CC(C)C(C)(CNC(c1cc(C2CC2)no1)=O)NC(c1cc(C(F)F)cs1)=O N1(C(c2c(C)cc(CNC(C3CCCO3)=O)o2)=O)CCCN(C2CC2)CC1 c1(N(C2C3CCC2CNC3)C2CC(=O)OC2)ncnc2ccc(F)cc12 CCC(C)C(O)C(=O)N(C)CC1(NC(c2cccc(O)c2F)=O)CC1 N1(C(=O)CC2CCN(C(C3(CO)CCOC3)=O)C2)CCC(=C(F)F)CC1 CC(C)(C)C(CO)C(=O)NCCCC1CCN(C(c2cc(Br)no2)=O)CC1 c1(C(=O)OC)ccc(C)c(CN(C(C(=O)CS(=O)(=O)CC2CCCO2)=O)C2CC2)c1 N1(C(C(C=C=C)C)=O)CC2(NC(=O)CN(C)Cc3ccccc3Cl)CCC1CC2 N1(C(C2C(C(C)C)OCC2)=O)CC(O)CC1(C)C(=O)NCC1CC(F)(F)C1 N1(C(CC(C)(C)F)=O)CCC2(CC1)CC2NC(c1cccc(OCC2CC2)c1)=O Cn1cc(C(N2CCCC(n3cc(CNC(=O)CO)nn3)C2)=O)n(C)c1=O c1(C(=O)NCCCOCCN(C)C(C23CCC2C3)=O)cc2cc(Cl)ncc2[nH]1 CC(CC(=O)NC1CC2(C1)CC2NC(=O)C(F)=C1CCCC1)C(F)(F)F C12(C(N(CC(CN(C)C(c3cc(CO)on3)=O)O)C)=O)CCCN1CCC2 Cc1ccc(O)c(NC(c2ccc(-c3ccc(F)c(F)c3)c(C)n2)=O)c1 C#CC1(C(=O)Nc2cn(C)nc2O)CCN(C(=O)C=CCCC)CC1 c1(CC(=O)NCCCNC(C2CCC(F)CC2)=O)c(Br)ccc(F)c1F c1(OC)c(Cl)nc[nH]c1=NCC1CCCCC1NC(=O)Cc1ccc(C)c(Cl)c1 CC(C)(C)C(C(=O)NCC(CO)NC(=O)CCC1CCCC1)N1CCOC1=O CCCCC(CN(C)C(C1CCN(C(c2ccnc(CC)c2)=O)C(C)C1)=O)CC Cc1cc(C#N)nc(N2CC(NS(=O)(=O)c3nccs3)C(C#N)C2)n1 N1(C(C(CC)COC)=O)CCCCCC1C(=O)NCC1CC12CCOCC2 C=C(C)CCCC(=O)N1CCC(O)(CNC(c2cccc(NS(C)(=O)=O)c2)=O)C1 C1(CNC(Cc2c(C)non2)=O)CCCN(C(=O)Cc2ncsc2Cl)CC1 C1(F)(C(=O)NCC2CCCN(C(CC(CC)OC)=O)C2)CCCCCC1 C(=O)(C(C)CCC(C)(C)C)N1CCC2(CN(C(C3OCCN(CC)C3)=O)C2)C1 c1(C(N2CCOCC(NC(C3CC(C)N(C)C3)=O)C2)=O)c(F)ccc(Cl)c1N C1(NC(C(C=C)(C)C)=O)CC2CCC(C1)N2C(c1c[nH]nc1S(N)(=O)=O)=O c1(C(=O)NC(C(C)NC(c2nc(C)n(C)c2)=O)(C)C)ncc(Br)cc1F CC1(C)CCCC(O)(C(=O)NC2CCN(c3nc(Cl)ncc3C(N)=O)CC2F)C1 c1(C(N(C2(CC(=O)N(CCNC(C(C)C)=O)C)CC2)C)=O)cc2cc[nH]c2cn1 c1(C(=O)NC(C2CCN(C(CSCC)=O)C2)C)c(Br)sc(C)c1C C1(CC)(NC(c2cncc(OC)n2)=O)CCCN(C(=O)C(C)OCC2CC2)C1 C1(CC(=O)NC(C(CC)(F)F)(C)C)SC2=NCCN2C1=O Cn1nc(O)cc1C(N1CCC(C(O)CNC(c2cncc(Cl)c2)=O)CC1)=O N1(C(C(C)OCC2CC2)=O)CC2CCC1C2NC(c1cncc(N)c1)=O N1(C(C2CN(C(=O)NC)C2)=O)CC2CCN(C(=O)CCn3nc(C)nc3C)CC12 C1(C(N(CCNC(C(CCC)F)=O)CC)=O)CNC(=O)C(C)(C)C1 N1(C(C2C3CCCOC23)=O)CCC(O)CCCCC1(F)F Cc1cccc(C(N2CCC(O)(CNC(C3CC3c3ccccc3)=O)C2)=O)c1O c1(NC(c2ccc(Cl)o2)=O)ccc2c(c1)CN(C(C1CC=CCC1)=O)CC2 C=C=C(C)CC(=O)N1CC(O)(C(C)NC(=O)CN2CCC(C)(O)C2)C1 N1(C(C2(CC#C)CCOC2)=O)CCC(CNC(=O)C(C)(C)C2CCC2)(OC)C1 c1(C(=O)NC(CCCC)CNC(=O)CCc2ccsc2)ccn(CC)c(=O)c1 C12(C(NOC(CC)C)=O)CCN(C(=O)Cn3cnnc3)CCC1C2 C(=O)(CCC(C)O)NCC(CNC(CC1C(C)CCC1)=O)O CC12CCC(C(=O)NC3CCC3CNC(=O)Cc3ccoc3)(CO1)C2 n1(CC(C)O)cc(C(=O)NC2CN(C(C3(C)C=CCC3)=O)CC2C)ccc1=O Cn1ncc2cccc(CC(=O)NCc3nc4cc(F)ccc4s3)c12 C1(NC(c2n(CC)cnn2)=O)CCC2(CC1)CC2NC(=O)C(CC)SC c1(C(N2CC(CN(C(C3C(COC)C3)=O)C)OCC2)=O)ccc([N+](=O)[O-])cn1 c1(NC(C(c2[nH]nnc2C)N(CCOC)C)=O)c(C)cc(C)cc1C c1(C(=O)NC(CNC(=O)C(O)(C(F)(F)F)C2CC2)CO)ccnc2ccncc12 N1(C(Cn2ncc(C#C)c2)=O)CC(NC(=O)COCP(C)(C)=O)CC(O)C1 C1(C(N(CCO)CC)=O)CCN(C(C2(C)CCSCC2)=O)CC1(C)C C1(C(=O)NC2COCCN(C(c3c(C)cno3)=O)C2)COc2cc(Cl)ccc2C1 c1(C(=O)NCCCOCCN(C(=O)C=C2CCCC2)C)coc2ccccc12 CCCCCCC(C)C(=O)NCCC(C)(C)NC(=O)Cc1ccc(C(N)=O)nc1 CCC(C(=O)N(CCCC(=O)NCC(C)(C)OC)C)n1cncn1 C(c1cccc(Cl)c1)=C(C)C(=O)NC1CCN(C(C2CCCCC2)=O)C12CC2 N1(C(c2c(CC)noc2C)=O)CC2CCN(C(=O)CC3CC(C)=NO3)C2C1 c1(C(=O)NCC2N(C(Cn3c(C)ncc3)=O)CCC2)cc(N)cnc1Br c1(OC)ccc(C)cc1CC(N1CC(NC(=O)CSCCOC)C2CC2C1)=O c1(C(=O)NC(CNC(C(C=C=C)C)=O)C)ccc2cnnc(O)c2c1 C=CCC(CC=C)C(=O)NC1CCCN(C(=O)COCC(F)(F)F)CC1 N1(C(C2N3C(C)CN(CC3)C2)=O)CCC2(CCN(C(=O)C3=COCC3)C2)C1 C=CC(C)C(=O)N1CC(CC(=O)NC2CC(N(C)C3CC3)C2)(OC)C1 c1(-c2ccc(C=C)cc2)cnn2cc(C(=O)N(C)C3CC3)cnc12 C1(N(C(C2CCC(=C)CC2)=O)C)CCCN(C(=O)CCOCC2CCCO2)CC1 c1(C(C(N2CCC(NC(C(C)(C)NC(=O)OC)=O)C2)=O)C2CC2)ccc(C)cc1 CC(O)CCCNC(c1sccc1CNC(=O)C(C)(C)C1CCCC1)=O C(=O)(C1=COCCC1)N(CCCNC(c1ccc(Cn2ccnc2)o1)=O)C1CC1 N1(C(=O)Cc2ccccc2O)CCC(F)C(NC(C2(O)CCCCC2)=O)C1 N1(C(=O)NCc2nc(C)sc2C)CCN2C(=O)CCC12C c1(CC)cc(C(=O)NCC2CC(O)CN2C(=O)CNc2ccc(Cl)cc2)nn1C N1(C(C(c2cccc(C)c2)=O)=O)CCCC(CO)(NC(=O)CCC=CC(C)C)C1 c1(NC2CC3CN(C(C(C)(F)F)=O)CC32)cc2nc(O)oc2cc1[N+](=O)[O-] CC(C)C(Cc1ccccc1)C(=O)N(CC(C)CNC(c1cnn(C)c1)=O)C C=CCCC(F)(F)C(=O)N1CCC(NC(c2cnoc2CC)=O)C(CC)C1 c1(C(=O)NC(C)C(CO)NC(=O)CC2CC=CC2)ccc(Cl)cc1F c1(NC(N2CC3CCCC3(CO)C2)=O)cnn2c1CCCC2 C#CC1CN(C(C2CC3CCC2O3)=O)CCN1C(c1cncc(NC)n1)=O N1(C(C2C(OC)(OC)CC2)=O)CCC2(C1)CN(C(=O)C(C)Sc1ccccc1)C2 Cc1cncc(N(c2cnn(C3CN(C(C)C)C3)c2)C(c2cccnc2Br)=O)n1 CC(C)C(C(=O)N1CC2CC1C2NC(c1cn[nH]c1)=O)N1CCN(C)CC1 C(=O)(CCC(C)S(C)(=O)=O)NC1CCN(C(c2ccc(C#C)nc2)=O)CC1O C(c1cccc(CO)c1)=CC(=O)NC(C(C)NC(C1CC12CCC2)=O)CO C(=O)(C1=CC2CCC1C2)NCCCCN(C)C(c1cc2ccncc2[nH]1)=O C1(NC(CCSc2nc(C)[nH]n2)=O)CN(C(C2CCOCC2)=O)CC12CCCC2 C(=O)(C(O)CC(F)(F)F)NC1C2C(C)N(C(CNC(c3cc(C)nc(O)n3)=O)=O)C1C2 C(=O)(CC1=CCOCC1)NC(CC)CN(C)C(c1ccccc1F)=O C1(CN(C(=O)CC2CCCC2C)CC)CCN(C(c2ccsc2C)=O)CC1 C1(NC(CCOCCC)=O)CC2(CCC(CNC(=O)CC(C)C)OC2)C1 N1(C(c2c(CNC(c3c(C)ocn3)=O)noc2)=O)CCC2(C)CCCC12 N1(C(C(C)N2CCCC2)=O)CCC(C(F)C(=O)Nc2ccc(C(=O)O)o2)C1 C(CC(O)CC(=O)NCCN(C(C1CC1C1CCC1)=O)C1CC1)SC C1(C(N(C2CCN(C(c3sccc3CC)=O)CC2)CC#C)=O)CCCSC1C c1(C(N(CCNC(C(CCOC)C)=O)CC2CC2)=O)cc(C(=O)OC)ccc1Cl C1(NC(C2CCSCC2)=O)C2CC1CN(C(=O)Cn1cncn1)C2 C1(C)(C(N2CC(COC)C2)=O)CN(C(=O)CCC2CCCO2)C1 C(CCCC(=O)NC1CN(C(=O)C=NOC)CC1C(F)(F)F)OCCC=C C(=O)(CCN(C(=O)COCC)C)OCC.C1CNC(=O)N1 c1(C(=O)NCC(C)(CO)NC(c2nc(COC)sc2)=O)c[nH]c2cc(C)ccc12 C12(C(=O)NC3C(NC(C(c4c(C)cncc4)C)=O)CC3)CCC(CC1)OC2 N1(C(c2n(CC#C)ccc2)=O)CC2C3CCC(C2C1)N(C(c1ccc(Cl)o1)=O)C3 C(=O)(C(=O)C(F)(F)F)NC(CCNC(C(C)C(C)c1ccc(F)cc1)=O)C N(C(=NCCF)NCc1ccnc(Cl)c1)CCNC(c1ccccc1)=O CC(C)CC(C(=O)NC1CCC(NC(C2(c3ccn(C)n3)CC2)=O)CC1)C(N)=O CCCCCCCCCC(C)(c1nnnn1C1CCOCC1)NCc1ccco1 CC1CCCn2ncc(C(=O)N(C)CCNC(c3c(Cl)ccc4c3OCO4)=O)c21 N1(C(c2cc(Br)cs2)=O)CC2CC2(CNCc2ccncn2)C1 C1(CNC(C(c2cccs2)NC(C=CC=CCC)=O)=O)(CO)CCN(C)C1 N1(C(CCOC)=O)CC(NC(=O)CC2SC(=N)NC2=O)C2CCCC2C1 c1(C(N2CC(CNC(c3c(OC)c(Cl)ccc3)=O)C2)=O)cccc2oncc12 c1(C(=O)NC2C(NC(c3cc(CCC)n(C)n3)=O)CCC2)ccnc(Cl)c1O CC(C)CC(C)C(=O)N1CCCCC1C1CCN(C(c2coc(C(F)F)n2)=O)C1 c1(OC)ccc(CNCC23CC2CN(C(c2ccnn2C(C)C)=O)C3)c(Cl)c1Cl C(=O)(C(C)(F)CC1CCCC1)N(C1CC(NC(c2cn(C(C)(C)C)nn2)=O)C1)C CCC(C)(C)C(=O)NC1CCCCC1NC(=O)Cn1nc(C)cc1C C1(CN(C(C(CC)N(C)CC)=O)C2CC2)CCN(C(=O)CCc2cnc[nH]2)CC1 CC(C)C(C(=O)N1CCCC1Cc1ccccc1Cl)SN(C)C(C12CCC1C2)=O C1(CCC)(NC(c2cccs2)=O)CCCN(C(C23CCCC2C3(F)F)=O)C1 C1(CNC(C2CC2C(F)F)=O)CCCCN1C(c1n[nH]c(C2CC2)n1)=O N=c1[nH][nH]c2cccc(C(N3CCC(NC(=O)CNC=O)C(F)C3)=O)c12 C#CC1(O)CC(C(N2CC(F)(CNC(=O)CC(C)n3cc(Br)cn3)C2)=O)C1 c1(C(=O)NC(C)C(CO)NC(c2cnc3n2CCS3)=O)cnc2c(c1)COCC2 c1(C(=O)NCCCCNC(c2c(OC)csc2)=O)cnc(C(N)=O)cn1 C(=O)(CCC(C)CN(C)C)N(CCC(N1CCC(C(=O)NC)C1C)=O)C N1(C(CN(C(C)=O)C2CC2)=O)CCC2CCC(NC(C3CC(C#N)C3)=O)C1C2 N1(C(CCN(C(CCC)C)C2CC2)=O)CCCC(NC(C2OCCO2)=O)C1 c1(Sc2cc(C(C)C)nn2C(=O)C(C)(C)C)cc([N+](=O)[O-])ccc1Cl C1(C(N2CC(C(=O)NCC(NOCC)=O)(SC)C2)=O)CC(=O)CCO1 C1(CNC(C2C(OC)C2)=O)COCCN(C(c2cn(C)cc2C(F)(F)F)=O)C1 C(C)(C(=O)N1CCC(CC(C)NC(=O)CN2CCNC(=O)C2)CC1)(C(C)C)OC N1(C(C(c2ccnn2C)NC(CNC(COC)=O)=O)=O)C2CCCC1CC(O)C2 N1(C(=O)CC2CC(F)(F)C2)CC(CNC(C2(C3CC3)CC2)=O)C2CC12 N#Cc1csc(CNC2CCCC2C(N2CC(O)C(O)C2)=O)c1 C1(OC)(CNC(=O)N(C2CC(c3ccc(Cl)cc3)C2)C)CS(=O)(=O)C1 CC1CCN(C(C2(CO)CCCO2)=O)CCN1C(C1(CCF)CCC1)=O C1(C(=O)NCCN2CCC(C)C2)(CNC(COc2cc(C)on2)=O)CC12CCC2 C1(NC(c2csc(C)c2C)=O)C2CC3C1C3C2C(=O)NOCCSc1ccccc1 CC(c1ccsc1)=CC(N1CCCC1C1(NC(C2C3CC4C(C3)C24)=O)CC1)=O Cc1nnc2n1CC(C(N1CCC(O)(Cc3ccc(O)cc3)C1)=O)CC2 c1(-c2n(C3CC(C)OC(C)C3)nc(C(F)F)n2)cccc2nc[nH]c12 Cc1nc2c(s1)CCCC2CNc1nn(C)c(C2CCCCC2)c1Cl CC#CCCCC(=O)NC1CCCC(CNC(c2cn(C)c(=O)cn2)=O)C1 C1(CNC(c2cnc3sccn23)=O)CN(C(C2CC3CCC(C2)C3)=O)CC12CC2 CC(C)C(CNC(=O)CC1(C#N)CC1)C(=O)NCCC1NC(=O)NC1=O C1(NC(c2c(-c3ccc(C)s3)c[nH]c2)=O)CCN(C(C2CS(=O)(=O)C2)=O)CC1C C(=O)(C1=CC2(CCOC2)C1)N1CC(=O)NCC1C(N1CC(CO)(CF)C1)=O N1(C(C(=O)NC(CNC(Cc2c(C(=O)OC)csc2)=O)SC)C)CCCCCC1 c1(C(=O)NCC2N(C(C(C)=C(CC)C)=O)CC2)cnn2cccc(C)c12 c1(C(C)C)ccc(C(=O)NCCN(C)C(C2CCC(F)(F)CO2)=O)cc1[N+](=O)[O-] c1(CNC(C2N(C(CC3(C=C)CCOCC3)=O)CC2)=O)c(OC)ncc(Cl)c1C N1(C(c2c(COC)cco2)=O)CCOC(CC(=O)NCC(C)(C)CO)C1 C(=O)(C#CC1CCCO1)NCCNC(c1ccc(=N)[nH]n1)=O.C12CN(C1)C2=O CCCCCCC(=O)NC(C)CCNC(=O)CCC(=O)NCC C1(N2C(=O)CCC2)COCC2(CCN(C(=O)C(N)CCCC(=O)OC(C)(C)C)C2)O1 C=CC1(NC(=O)CC2CCCC2NC(c2ccncn2)=O)CCCC1 C(=O)(CCC(=O)N(C(C)(C(=O)NCc1ccnc(Cl)c1)C1CC1)C)NCC C(C(=O)NCC1CCCO1)(C(C)Cc1ccsc1)N(C1CCN(C)CC1)CC C1(NC(C2C(OC)CCC2)=O)CC2CCC(C1C)N2C(C1COC(C)C1)=O Cc1nc(C)c(CNC(=O)C=CC(C)NC(=O)C(C)N=[N+]=[N-])s1 CCC(COC)C(=O)NC1C2CC(NC(c3ncccc3OC)=O)CC12 c1(C(=O)NC(c2ccc(OC)cc2)C2CCCC2)ccc(Cl)nc1O C=CCC(C)(C)CC(=O)NCC(C)NC(=O)CCC1CCN(C)C1 Cn1cc([N+](=O)[O-])cc1C(N1CC(CNC(=O)CCS(N)(=O)=O)C(C)(C)C1)=O N1(C(C2(CCC=C)CC2)=O)CC(CNC(c2cc(N)c(Cl)cn2)=O)C(C)(C)C1 N1(C(c2c(OCC#C)nccc2)=O)CCN(C(C2CC=CCC2)=O)C2COCC12 CC1C(NC(=O)C(C)C(C)(C)C)CC2CCC1N2C(=O)CC1CC(C)(C)CO1 c1(SC)cc(C(=O)NC(C)C(CO)NC(c2cn(CC(N)=O)nn2)=O)oc1C C1(CC)CCOCCN1C(=O)C(CNC(c1ccc(=O)n(C)c1)=O)OC N1(C(CC(C)(C)SC)=O)CCCOC(CCNC(c2ccc(C)cn2)=O)C1 c1(CC)ncc(C(=O)NC(CNC(=O)CSC)C2CC2)[nH]1 C1(C(C(=O)NCc2ccccc2)N(C23CC(C2)C3)C)CC2(CCC2)C1 C(CC1CCC1)(C(=O)NC(C)Cc1cnc[nH]1)NC(CCSCC)=O c1(C(C)C)ccccc1OCCC(=O)NCCC(C)NC(c1cn(C)nc1O)=O c1(OC)nc(N2CCCC(NC(=O)C(c3cccn3C)=O)C2)ncc1F c1(C(=O)NCC2C(CNC(CN(C3CC3)CC)=O)C2)cc(F)c2ncccc2c1 C=CC1(CC(=O)NC(C)CCNC(=O)CN2CC3CC3C2)CCOCC1 C1(C)(C(=O)NCC(CNC(C2(COC)CC=CC2)=O)(C)O)COC(C)(C)CO1 N1(C(C)=O)CCN(CC2(OC(C(C)=CCC)=O)CC2)CC1.c12ccc(cc1)o2 CN1CCC(C(=O)NC2(CN(C(=O)CCC3CC3(Cl)Cl)C)CC2)C1 C1(NC(C2CC(OC)C(OC)C2)=O)CN(C(=O)Cc2c(C)noc2C)CCC1O N12CCC(C)(CC1)CC(=O)OC1CC(C1)C2=O.n1(CC)nnnc1COC(C)(C)C Cc1cccc(C=CC(=O)NC2CCCN(c3cnccn3)C2)c1 CC1CN(C(=O)CCn2cccn2)CC(CCNC(C2CN(C3CCC3)C2)=O)O1 C(=O)(CCC(=O)N1CCCCC1C1CCCN(C(C2(C)CC2(Cl)Cl)=O)C1)NCC Cc1nc(NCC(c2nccs2)C)cc(N(C)CC2CCCCO2)n1 c1(OC)cccc(F)c1C(C)NC(=O)NCC1SCCN(C)C1.c1ccccc1 Cc1c(Cl)nc(C2CC2)[nH]c1=NCC1CCN(C(=O)C=Cc2nccs2)C1 Cc1cc(NC(=O)CC2CCCCC2NC(C2CN3CCC2C3)=O)ccc1O c1(C(=O)NCC(CCNC(CC2C(CC)C2)=O)(C)C)ccc2c(c1)OCO2 N1(C(c2c(OC)nn(C)c2Br)=O)CC2(CCCCN2C(C2CC2C)=O)C1 C#Cc1ccc(CC(N2CC(C(O)C(=O)NC(CC)C(=O)NC)C2)=O)cc1 C(=O)(C(O)(CN(C)C)C(F)(F)F)NCC1CCN(C(C(CC)(C)COC)=O)CC1 N1(C(C(CC=C)(F)F)=O)CCCC2(C1)CN(C(=O)C(n1ccnc1C)C)CCO2 CN1CCC(OCc2cn(CCCNC(C3CC(CF)C3)=O)nn2)CC1 CCC(C)(CNC(C1CCCN(C(=O)COCCOC(C)=O)C1CC)=O)C(N)=O C1(N2CCCCC2)(CCN2CCCC2)CCCCC1.CC(CCCc1cccnc1)NC=O c1(CC)ccnc(C(=O)NC(CC2CCCC2)C(=O)NCC(O)C(C)O)c1 c1(C(=O)NC(c2ccccc2)C(=O)OC(C)C)noc2c1CN(C(C)C)CC2 C1(CNC(CCC#C)=O)CN(C(C2CCCN2Cc2nnn(C)n2)=O)CC12CC2 C1(NC(CC2(C)CC(F)(F)C2)=O)CCN(C(=O)C(O)C(F)(F)F)CC12CCC2 C1(C(=O)NCCOC2CN(C(C3CCC=CCC3)=O)C2)CCCC2CCCN12 N1(C(C=C(C)C)=O)CCCC(C)(C)C1CNC(C1(CO)CC1)=O.S(=O)(=O)(C(F)F)N C(c1cnc(OC)nc1)=CC(=O)NC(CN(C(c1ncoc1C)=O)CC)C C1(COC)(CNC(C2CC(F)C2)=O)CCN(C(=O)C=CC2(C)COC2)C1 NS(=O)(=O)C1(c2cn(CCNC(C3(O)CCSC3)=O)nn2)CC1 C1(C(=O)NCC2(C)N(C(C3CN(C(C)=O)C3)=O)CCC2)CC2(C1)CC(F)(F)C2 c1(C(N(CC(CC)NC(C2CC(F)(CO)C2)=O)C)=O)c(C)nn(C2CC2)c1Cl c1(C(N2C(CNC(CCCOCCC)=O)CCC2)=O)ccc(COC)cc1OC C1(C(=O)NCC(C)(C)SC)CCN(C(=O)C=CC2(C)COC2)C(C)C1 C(=O)(CC(C)(C)C)N(CCCNC(=O)CCC=CC(C)C)CC c1(CCC)cc(C(=O)NC2CC(F)(CNC(c3sccc3CC#N)=O)C2)n(C)n1 c1(NC(C2CCN(C(=O)CC34CCC(CC3)C4)C2)C)[nH]c(=O)n(C)c(=O)c1C#N c1(C(=O)NC(C(C)NC(c2c(C)nsc2)=O)C(C)C)nccc(N)c1Cl C(c1nnn(C)n1)=CC(=O)N(C(CCNC(CCC=CC(C)C)=O)C)C N1(CC(=O)NC(C)C(C)NC(c2cnccn2)=O)CCS(=O)(=O)CC1 C(C)(C)(CN=c1nc(C#N)[nH]cc1Cl)NC(C(C)CC1CCCC1)=O C(=O)(C1=NOC(C(=O)NC23C=CC(CC2)C3)C1)NC1(C)CC(CO)C1 c1(NC(=O)OC(C)(C)C)ccoc1C(=O)NCCCCCNC(C12CC(CO1)C2)=O N1(c2snc(SC)n2)CC2CCC(NC(=O)C#CC3CCCCO3)CC2C1 N1(C(C2CC(=C)CN2C(c2ccc(Cl)c(C#N)c2)=O)=O)C2CCCC1COC2 C1(C(=O)NCC2CC(CNC(=O)C(N3CCNC3=O)C)C2)(CC)CC(C)(C)C1 C1(CCS(=O)(=O)N(C2C(C)C2)C)CCC2(CC1)CC2 C1(CC(=O)NC(CNC(C(C)(C)CF)=O)C2CCC2)CCOC(C)(C)C1 c1(NC(C)=O)ccc(F)c(NC(=O)NC2CC(c3ccc(F)cc3)CC2O)c1 S(=O)(=O)(c1ccccc1)Nc1c(C(=O)OCc2n(C)nnc2)cccc1 Cc1cc(NC2CCCN(CC(N)=O)C2)ncc1S(=O)(=O)N1CC=CCC1CO C1(NC(c2n(CC#C)ccc2)=O)CCN(C(=O)C(O)Cc2ccccn2)C12CC2 c1(C(=O)NCC2CC(C)(C)N(C(c3cnsc3)=O)C2)c(N)ccc2nccnc12 N1(C(Cc2c(C)nn(C)c2)=O)CC2CCC1C(NC(=O)C(O)Cc1cnc[nH]1)C2 c1(OC)ccc(C(=O)NC2(CNC(=O)C=CC3CCCO3)CCC2)c(F)c1N N1(C(CC(COC)COC)=O)CCc2nc(CNC(=O)C(O)CCSC)sc2C1 C(C(C)(C)C(=O)N1CCOC(C(C)NC(c2[nH]ccc2COC)=O)C1)OCC C12(CNC(c3ccccc3F)=O)CCCC1CN(C(c1cnns1)=O)C2 N1(C(C(C=C)(C)CCOC)=O)C2CCC1CN(C(c1c(N)cccc1F)=O)CC2 CC1CCCC1C(=O)NC1(CNC(c2ncoc2Br)=O)CCCC1 C1(CC)C(=O)NCCCN1C(C1(CNC(=O)C(COC)N(C)C)CCCC1)=O c1(C(=O)NC2C(C)(CNC(=O)CC3(C#N)CC3)CCC2)occ2c1CCCC2 N1(C(COCC#C)=O)CCN(CC(=O)NCCO)CC1.CC O=C(C1=C(Cl)CCOC1)NCCN(C(c1cnc(O)o1)=O)Cc1cccc(Cl)c1 c1(C(=O)NC(CNC(CCCOCCOC)=O)(C)CO)cccc(N)c1 C1(C(=O)NC(C2CCOCC2)C)CC2CCC1N2C(c1c(Br)cncc1Br)=O CC(C)CC(C)CC(=O)N1CCOC(C(C)NC(c2cnc(Cl)[nH]2)=O)C1 C1(C(=O)NCC2N(C(CC(C)NC(=O)C3CC3)=O)CCC2)CCC(F)(F)C1 C1(N(C)C(=O)C2CC2)CCCN(C(=O)CC2CC23CC3)C1 N1(c2ccc(S(=O)(=O)N(CCCC(C)C)C)cn2)CCCC(C2CNC(=O)C2)C1 C1(N(C)C(=O)NC(C(=O)OC(C)(C)C)C2CCC2)(CO)CCCOC1 C1(C(=O)OC)CN(C(c2nn(C)cc2C)C(=O)NCCSC)CCN1C(C)C CC(F)(F)CCCC(=O)N1CCCC(CNC(C2(C)CC=CCO2)=O)CC1 C(C(CC(F)(F)F)NC(=O)Cc1cn(C)nc1C)NC(c1c(OC)cncn1)=O C1(CS(NC2=NCC(C)S2)(=O)=O)CCN(C)C(C)(C)C1 N1(C(CCC#CC)=O)CC2CN(C(C3CCN(Cc4ccccc4)C3)=O)CCC12 c1(SC)ccc(-c2nc(CCC(F)(F)F)nn2C(C)C(C)C)cc1 C(N=c1[nH]c2ccc(O)cc2s1)C1CCCC(NC(C2CC23CCOC3)=O)C1 C=CCCCC(C(=O)N1CCC(F)(CF)C1)NC(=O)CSC CC(C)CCC(=O)N1CC2C(NC(c3cn(C(C)(C)C)cn3)=O)C2C1 C1(CC(=O)NC2(CNC(C3(CCC)CCC3)=O)CCC2)OCCC1C c1(C(N2CCN(c3c(Br)cnc(SC)n3)C(C(C)C)C2)=O)c(Cl)cnc(Cl)c1Cl n1(CC(=O)NC2CC3(C2)CN(C(c2nc(Br)c[nH]2)=O)C3)ncc2cccnc12 C1(NC(c2c(Cl)cn(C(C)(C)C)n2)=O)CC2CCC(C1)N2C(C1CCCOC1)=O N12C(CCC1C(=O)O)C2=O.n1(C(C)C)ccc([SH](CCCOC(C)(C)C)N)n1.C(=O)O C1(C(C)(C)O)CCN(C(C2CCCC2NC(=O)CC#N)=O)C1 c1(OC(C)(C)C)cc(F)cc(C(=O)NC2(n3cnnn3)CC2)c1N c1(NC(CC2CC(NC(C=CC=CC)=O)C2)=O)cc(OC)cc(C)n1 Cc1nccc(C(=O)NCC2CCCC2C(N2CC(CCO)C2)=O)c1N C1(c2n(CCC)nnn2)(NC(C)Cc2ccco2)CC(C2CCCCC2)C1 CC(C)C(C)(CNC(c1ccc(C2COCCN2C(=O)C=CCF)n1C)=O)OC N1(C(CS(=O)(=O)NC)=O)CC(CNC(C2CCCCCCC2)=O)OC2(CCC2)C1 c1(C(C)(C)C)n[nH]cc1C(N1CC(O)(CNC(C2(C3CC3)CCCO2)=O)C1)=O C(=O)(CCC(CC)OC)N1CC(NC(c2c(CC)non2)=O)C1 Cc1cccc2[nH]cc(C(=O)N(C3CCN(C(=O)C4=CCCS4)C3)C)c12 c1(OCC)cccc2c(=O)c(C(=O)NCCN(C)C(C3CCC(C)C3)=O)c[nH]c12 C1(C(C2CCOCC2)C(=O)NC)CCCCN1CCc1ccc(OC(C)C)cc1 c1(CCN(C2CC(c3ncc[nH]3)C2)C=O)ccccc1OC(c1c(C)ccs1)=O C1(CC(=O)NCC(C(=O)OCC)(C)O)CCC2(CCC2)CO1 c1(C(=O)NCCN(CCC)C(c2cc(C(N)=O)c[nH]2)=O)csc(-c2cnc[nH]2)n1 C(=O)(CP(=O)(C(C)C)C(C)C)N1CC(CNC(C=CCCC(C)C)=O)C(O)C1 C#CC1(C(=O)NCC(c2nccs2)C)CN(C(=O)CC2C=CCC2)C1 c1(C(N2CCC(CCNC(CCSCC)=O)C2)=O)cc(N(C)C)ncn1 C(F)(F)(C(F)(F)F)OCC(=O)NCC1CCN(CCN2CCOCC2)C1 C1(NC(c2cc(C)cc(F)c2)=O)CC2CCC1CN2C(c1csc(C)c1C)=O c1(CC(=O)NCCN(C(CC=CC)=O)C)cc(C)no1 c1(CN(CC(CC)O)CC)cccc(-c2cccc(CC3CCC3)c2)c1 c1(CC(=O)N(CC(C)CNC(C2CCC2)=O)C)cc2c(cc1Br)OCO2 N1(C(CSCC)=O)CC2CC(NC(=O)C(C)NC(=O)NCC)C2C1 c1(C(N(CCCN(C)C(C2(C3CCCO3)CC2)=O)C)=O)ccoc1Br c1(OC)cccc(C2CCN(Cc3cccc(SC)c3)C2)c1OCC1CCC1 N1(C(c2nc(CC)sc2)=O)CC(CNC(=O)C(C)CN(C)C)OC(C)(C)C1 N1(C(C2(C=C)CC2)=O)CCCN(C(=O)CSCc2cscn2)CC1 C(=O)(C(O)C(F)(F)F)NC(C1CCN(C(C(C=C)CC)=O)C1)(C)C C1(C2CC2)(NC(CC(=O)OC(C)(C)C)=O)CCN(C(=O)Cc2ccsc2)CC1 N1(C(CC=CCC)=O)CC(F)(CNC(c2cnn(C3CCCCC3)c2)=O)C1 N1(C(C2COCC(C)O2)=O)CCC=C(C(=O)N2CC3CC2CO3)C1 C(CCC)(C(=O)NC(c1nc(=O)o[nH]1)C)NC(C(CC)OCC)=O c1(C(C(=O)NC2CC2CNC(C2C=CCS2)=O)OC(C)=O)ccccc1 C1(NC(=O)OC(C)(C)C)CCCCC1C(N1CCC(CCNC)C1)=O C12(C(N3CCCCC(n4cc(CS(CC)(=O)=O)nn4)C3)=O)CCC(F)(CC1)CC2 N1(C(CCC2C(C)C2)=O)CCC(CC(=O)N(c2cnc(F)nc2)C2CC2)CC1 Cc1c(Cl)ccc(C(=O)N(C23CCC(CO)(C2)OC3)C2CC2)c1O C(=O)(CCCNC1CCOCC1)NCC1C(CC(=O)N(CC(C)(C)C)C)C1 C(N=c1cc(NCCOCCF)nc(CC2CC2)[nH]1)C1C(c2cccc(C)c2)C1 C(=O)(C(C(CC)CC)OC)NCC(CC=C)C(=O)N1CCCC(C#C)C1 N1(C(c2cnc[nH]2)=O)CC2(NC(C3CCN(c4ccncc4)C3)=O)CCC1C2 C1(C)(C(N2CC3C(NC(C(C)NC(=O)OC)=O)(C3)C2)=O)CCCCCC1 Nc1ccc(Br)cc1C(N1CCC(CF)(NC(=O)CCc2cnc[nH]2)C1)=O CC1CCCN(C(=O)OCc2cccc(F)c2)CC1N(C)Cc1ccccc1 Cc1c(Cl)ccnc1C(=O)NC1CC(N(C)C(C2CCCCC2(C)C)=O)C1 N1(C(CN(C(=O)C(C)COCC)CCC)=O)CCc2c(nnn2C)C1 C1(C(=O)NCC2(C(N3CCC(CC4CC4)C3)=O)CCCC2)CC12CCOCC2 c1(OC)cccc(C(N2CC(CNC(c3snnc3C(C)C)=O)CC2C)=O)c1N C1(CN(C(C2CCN(C)C2CC)=O)CC)CCN(C(C2(O)CCC2)=O)CC1 Cc1nc(NCCC2CCCCC2C)cc(N2CCNC(=O)CC2)n1 C1(C(=O)NC2CCC(OCCOC)C2)COCCC1NC(=O)C(=O)C1CCCC1 CS(=O)(=O)CCCC(=O)N1CC2CCCC2(CNC(c2cc3cscc3s2)=O)C1 c1(OC)noc(C(=O)NC(CNC(c2ccn(C(C)C)n2)=O)C2CC2)c1Br.C1CC1 CC1(C)CC(C(=O)NCCC2CC(F)C2)CCN1C(c1cc(C#N)c[nH]1)=O C1(CC(=O)NC(c2cn(C)nn2)CNC(C(=O)NC(C)C)=O)COCC(C)(C)O1 CC(C)(C(=O)N1CCC(C2CCCN2C(=O)C=Cc2cc[nH]c2)C1)N1CCCC1 c1(C(=O)NCC(CCNC(c2cc(C(C)(C)C)on2)=O)O)cc2cccnn2c1 c1(C(N2C(C)CC(NC(C3(C=C)CC3)=O)C2)=O)ccc2cccc(Cl)c2n1 C12(NC(c3c(OC)ncc(Cl)c3)=O)CCN(C(=O)CN(C)C)CCC1C2 N1(C(c2cc(C(C)C)nn2C)=O)CC2CCC2(CCNC(=O)CNC=O)C1 C(=O)(C(C(C)C)NC(N)=O)NCC(C(C)C)NC(=O)C(=O)Nc1ccc(Cl)cc1 CC1CN2CCN1C(C(N1CCCC(CCNC(C3CCC(=O)N3)=O)CC1)=O)C2 N1(C(c2ccnc(C)c2O)=O)CC(CNC(c2ccoc2Cl)=O)OC2(CCC2)C1 C12(C(=O)NCc3c(C(=O)NC(CC(=O)OC)C)cco3)CCC(CC1F)C2 N1(C(c2cc(C)no2)=O)CCCC2(CNC(C3CCCC3)=O)CC12 C12(C(=O)NCC(C)C3CCC3)C(NC(c3cnco3)=O)C3CC1C2C3 C1(NC(CCSC)=O)COCCN(C(c2cccc(F)c2SC)=O)C1 C1(C(N2CC3(CN(C(CSCC=C)=O)C3)C2)=O)CCc2n[nH]cc2C1 CON1CCC(C(N2CC(N(C)C(c3nn[nH]c3Cl)=O)C(F)C2)=O)CC1 C12(NC(CCCc3onc(CC)n3)=O)CCN(C(=O)C3=C(Cl)CCC3)CCC1C2 C1(C(CNC(COCC(C)C)=O)(C)C)CCN(C(=O)CCC2CCCCO2)CC1 C1(CNC(C2C(C)CC2)=O)CC12CCN(C(=O)C(C)(F)c1ccccc1)CC2 CC(CCNC(=O)C(O)C1CC1)N(C(=O)CNC(=O)NC1CC1)C C12(C(=O)Nc3cccc(CC)c3)CCCC1CCN2C(C1CCC1C#N)=O C(=O)(C1SCCc2sccc21)NCC(C1CCC1)NC(C(COC)(C)C)=O CC1C(=O)NC(=O)CN1C(C1(NC(C2CCCC2C2CC2)=O)CC1)=O c1(C(=O)NCC2C(NC(CN(C)CCO)=O)CCC2)ccc(Cl)c(F)c1 c1(C(=O)NC(CCNC(C(CC)Cc2ccccc2)=O)C)cc(N)c(F)cc1C N1(C(c2nc(C)[nH]n2)=O)CCC(C2CCCN(C(C34CCOC(C)(C3)C4)=O)C2)C1 Cc1cc(C(=O)NCC(C)NC(=O)C(C)n2cccn2)ncc1N N(C(=NCCC1=CCOCC1)NCCF)CC(c1ccc(F)cc1F)C N1(C(c2c(CC)cccc2)=O)CCN(C(c2cc(SC)oc2C)=O)C(C(F)F)C1 C(C1=NOC2(CCC2)C1)NC(C1(C#C)CCN(C(=O)C(C=C)OC)C1)=O C1(c2ccccc2)(NC(c2ccc(-c3nn[nH]n3)o2)=O)CCCO1 Cc1cc(C(=O)NCCC(C)(C)NC(c2ncc(F)cn2)=O)cc([N+](=O)[O-])c1O c1(C(CC)=O)cc(C(N2CC(CCNC(=O)CNS(C)(=O)=O)C2)=O)ccc1F N1(C(C2(C(C)(F)F)CCOCC2)=O)CC2CN(C(=O)Cc3cncnc3)CC2C1 C1(NC(c2c(C)cc(C)cc2Cl)=O)CC12CCS(=O)(=O)CC2 C(=O)(CS(=O)(=O)CCOC)NC(C1CCN(C(C=CC(=O)OCC)=O)C1)(C)C N1(C(C2C(NC(C3CCN(CC)CC3)=O)CCC2)=O)CCCC(C#N)C1 c1(-c2ccn(C)n2)nc(CC2CCC2)n(C2CCOC2C)n1 N1(C(CC2CN(C(COCC(=O)NC)=O)CC2C)=O)CCC2(CC(CO)C2)C1 N1(C(CC2(C)CC2(Cl)Cl)=O)CCC2(CC1)CC2CNC(=O)CCCN=[N+]=[N-] N1(C(c2c(C)cc(F)s2)=O)CC2CCCC1C2CNC(=O)CCn1ccnn1 c1(C(=O)NCC2N(C(C(C)CC3CC3)=O)CC2)ccc(F)c2[nH]ccc12 C1(CC=C)(NC(=O)CC2CCCOC2)CCN(C(c2coc(C3CCC3)n2)=O)C1 C(CC(C)(C)CC(=O)NC(C)CN(C)C(c1cncc(C(F)F)c1)=O)OC c1(C(N)=O)ccc(-n2cc(CNC(N3CC(n4ccnn4)CC3CO)=O)nn2)cc1 Cc1cccn2ncc(C(N3CCCC(NC(=O)CN4CC=CC4)CCC3)=O)c12 c1(C2C(CC(=O)NC3CCCC3)C2)ccccc1.C1C(=O)NCC(C2CC2)N1C Cc1cc(C(=O)NC2COCCN(C(c3cnc(N(C)C)o3)=O)C2)c(N)c(Cl)c1 c1(C(N2CCCC(C)C2CCNC(=O)CC#N)=O)c2c(nn1C)CCSC2 N1(C(c2c(Br)cn(CC)n2)C(=O)NC2CCC2)CCCC2(C1)CN(C)CCN2C c1(C(=O)NCC(C2CCC2)NC(C2(Cl)CC2(F)F)=O)cncc2c(O)nccc12 CC(O)C(C(=O)NCCN1CCN(C(=O)COCc2ccncc2)CC1)N(C)C C1(C(=O)NCC(=O)OCC)CC(O)CN1C(C1(c2ccccc2)CCC1)=O N1(C(=O)NCCCNc2n(C)ccn2)CC(C(F)(F)F)Cc2ccccc21 c1(C(C)(C)C(=O)NCC2CCCCN2C(C2(F)CCOC2)=O)cccc(Cl)c1F Cc1nn(C)c(=O)c(C(N2CCN(C(c3ccc(N)cn3)=O)C(C)C2)=O)c1C Cc1c(C(=O)NC(C(=O)NC2CC2CC(C)(C)C)C2(O)CCC2)ncn1C C1(NC(CC(C)(C)N(C)C(C2(C#N)CC23CCC3)=O)=O)CCCCC12CCC2 C1(NC(=O)CSC2CC2)CCC(O)CN(C(C2CC3CC(=O)C2C3)=O)C1 c1(CC)cc(C(N2CCC(OCCNC(c3cc(SC)c(C)o3)=O)C2)=O)ccn1 CC(CC(=O)N1CCC(N=[N+]=[N-])(C(N2CC3CCC3(CO)C2)=O)C1)C(F)(F)F Cc1nc(CC(C)C)c(NC(=O)CC2CN(Cc3cn(C)nn3)CCO2)s1 CC1CC(C(=O)NCC2=CCCCC2)CN(C(=O)Cn2cc(Cl)cn2)C1 CC1(C)C(N(C(c2nc(Br)cs2)C(=O)NCC2CCOCC2)C)C1(C)C c1(C(N2CCC(C(=O)NCCC(=C)CNC(C)=O)C2)=O)cn2cc(Cl)cnc2n1 C1(C(N2CCN(C(=O)CC3(CO)CCC3)C(CO)C2)=O)CCc2c[nH]nc2C1 CC(O)C(F)(F)C(=O)NC1(C)CCC(NC(=O)CCOc2cccnc2)CC1 N1(C(C(c2cccnc2)C)=O)C2CCC1CN(C(C1CCNC1C)=O)C2 c1(SC)cncc(C(=O)NCC(C)(C)OCCNC(=O)Cc2cnccc2C)c1 N1(C(C=C(C)Cl)=O)CCC2(CCCN2C(c2ccc3oc(=O)oc3c2)=O)C1 C(=O)(CC(F)F)NCC(C1CCCN1C(=O)CCc1cnc(C2CC2)o1)(C)C C(c1ccccc1F)=CCC(=O)N(CC(C)O)CCNC(C(C=C)OC)=O Cc1nc(C(=O)NC2(C3CN(C(C45CC(CO4)C5)=O)C3)CC2)ccc1C#N C1(c2nnnn2C2CCC2)(NCCOc2cccc(OC)c2)CCC(C)SC1 C(c1ccc(C(C)C)cc1)=CC(N1CCC(CCOC)(NC(CCSC)=O)C1)=O c1(OC)ccc(OCC2CC2)cc1.c12ccc(cc1)CNS(=O)(=O)C2 C#CC1(NC(C2CC(=C)CCN2C(c2ccc(F)s2)=O)=O)CC2CCCC12 C(N=c1nc(Cl)[nH]c(CC2(CCOC)N=N2)c1C#N)c1n(CC)ncc1 C1(NC(C(C2CCC2)OCC)=O)C2CC(CN(C(c3ccns3)=O)C2)C1CO n1(C(CC)NC(=O)C(c2cc(F)ccc2F)CN)cnc2ccccc12 c1(C(=O)NCC(C)CNC(C2(S(N)(=O)=O)CCC2)=O)ccn2ncnc2c1 C(=O)(C(O)C(C)c1ccccc1)NCCNC(C(c1n(CC)ccn1)(F)F)=O C(C1CCCCCC1)=CC(=O)NCC=C1CCN(C(C2C3CC4C(C3)C24)=O)C1 c1(-c2nc(C(CC)C)nn2CC(C)(C)C)cnc2c(c1)CCOC2 CC(C)CCC(=O)N(C1C=CCN(C(=O)C=CSc2ccccc2)C1)C1CC1 C1(N(C(CNC(C=COCC)=O)C)CCOC)CCCNS1(=O)=O C1(C(C(=O)N(CC(C)(C)NC(C2CC(C)C2)=O)C)OC)CC(C)(C)C1 n1(CCC#C)c(N2CCN(C(c3ccccc3)C)CC2)nnc1-c1cccn1C N1(CC(=O)N(C2(C)CN(C(=O)C(C(C)C)C3CCC3)C2)CCN)CCCC(C)C1.CO N1(C(c2ccc(C)s2)=O)CC2(CC(CNC(c3ccnn3C(C)(C)C)=O)C2)C1 N1(C(c2nnc(CC)s2)=O)CCC(C)(NC(C2CCC(=O)N(CC)C2)=O)CC1 c1(C(=O)NCC(CNC(C(COCC)(C)C)=O)O)ccccc1C#CC1CC1 CC12CC(C(=O)NCC(C3CC3)NC(C3CC4C=CC3C4)=O)(C1)C(C)(C)O2 C1(COC)(NC(=O)CCCCN2CCCC2)CCN(C(=O)C(F)(F)C2CC2)CC1 Nc1cc(C(=O)NC2CCC2CNC(=O)CCc2cscn2)nc2ccccc12 c1(C(N(C2CCN(C(Cn3ccc(C)n3)=O)CC2)C)=O)cnc2n1CC(C)CC2 C=C(C)CC(C(=O)NCCNC(C1(F)C2CCCCC12)=O)NC(C)=O c1(C(N2C(CNC(CC3C(C)(C)C3(C)C)=O)C=CC2)=O)cc2n(n1)CC(F)C2 c1(C(=O)Nc2cnccc2I)cc2cc(-c3ccc4oc(O)nc4c3)ccc2[nH]1 C1(C(CC)=O)(NC(c2nnc(C3CC3)s2)=O)CCOCC1 C(=O)(CC(C)NC(c1cnn(CCNC(=O)C(C2CCC2)OC)c1)=O)NCC N1(C(CCc2cc(C)on2)=O)CCCCC(CNC(=O)CSc2ccccn2)C1 N1(C(COC)C)CCN(C(c2cnc(CC3CCC3)s2)C(=O)NCCSC)CC1 C1(C(=O)NCCNC(N(C)C)=O)CCCN1C(=O)CN1CC2CC2C1 C12(C(=O)NC(CC(C)C)CNC(=O)C=CCO)CC(N=[N+]=[N-])C1C2 N1(C(C2(C)CCN(C(=O)Cc3ncccc3F)CC2)=O)CC2CCC(C1)C2C#N c1(C(=O)NC2(C)CCN(Cc3onc(CCC)n3)C2)cc(Cl)ccc1OCC N1(C(c2nnc(C)s2)=O)CCOC(CC(=O)Nc2nccnc2Cl)C1 CC1(C)CC(C(N2CCN3CCC2C3)=O)CN1C(=O)C=C1CCC1 C1(C(N2CC(NC(CCC(CC)OC)=O)C2)=O)CCn2ccnc2C1 CC1CCCC(C(=O)NC(CCN(C)C(C2(C)CC(F)(F)C2)=O)C(C)(C)C)CC1 c1(C(=O)NCC2C3CCCC2N(C(c2ccno2)=O)C3)ccc2c(c1)COB2O c1(CC(=O)NCC(C)CNC(C2CC23CC3)=O)cnn2c1OCCC2 c1(OC)cc(C(=O)N(C)CCN(C(=O)C(C)(C)N(C)C)C(C)C)c(N)c(C)c1 c1(OC)cc(C)cc(C(=O)NCC2C=CCN2C(c2c[nH]cc(C)c2=O)=O)c1C N1(C(C2CCCS(=O)(=O)C2)=O)CCN(C(=O)COCC(F)F)C2(CCC2)C1 Cc1ccc2c(NC(=O)COC(=O)CCC3CCCCC3)csc2c1 C(=O)(CC(O)CCCC)NC1CCCC(CNC(C2(C#C)CCCC2)=O)C1 N1(C(C(C)=CC)=O)CCN(C(C23CCC2CC3)=O)C(CCCC)C1 CCCCC(C(=O)N1CCC(CO)(CNC(=O)CCCC(N)=O)CC1)N(C)C CC1CCCC(N=c2[nH]c(=NCCN(C)C)c3[nH]ccc3[nH]2)C1 N1(C(C(C(C)O)OC(c2ccc(SCC#N)o2)=O)=O)CCc2sccc2C1 c1(C(=O)NCC(CC(=O)NCCCN(CC)CC)O)ccc2cc[nH]c2n1 N1(CC(=O)N(C(C)CNC(=O)CCCS(C)(=O)=O)CC)CCCCC(O)C1=O C=CCC(F)(F)CN(C(=O)C(C1CCCO1)NC(c1ccc(NC)cc1)=O)C C(=O)(CCCCCn1cnnn1)NC12CN(C(C3(CC)CCCCC3)=O)C(C1)C2 c1(C(=O)NCC(=C)CCNC(=O)COCc2cc(C)no2)ccccc1C(C)C Cc1nc(C(C)C)cc(CN(CCNC(=O)CC2CCC3(CCC3)O2)C2CC2)n1 N1(C(C2CCC(=O)N2)=O)CCC2(CC1)CC2(C)C(N1CCC2CCC12)=O N1(C(c2c(CC)n(C)nn2)=O)C2CCC1CN(C(C1CC13CC3)=O)CC2 c1(C(N(C)CCNC(=O)CCc2cnc[nH]2)=O)cnc2c(F)cccn12 CC(C)CCCCCC(=O)NC1CCCN(C(=O)Cc2cc(F)cc(Cl)c2)C1C C1(C(=O)NCCC2CC(NC(C(N)=O)=O)C2)(Cc2cccc(F)c2)CCCCC1 C1(OCC)CCC(CC(=O)NC2CC(C)N(c3nnc(C(N)=O)s3)C2)CC1 c1(CC)nc2ccc(Cl)cn2c1C(=O)NC(CNC(C1CC1C#N)=O)C(C)(C)C N1(C(=O)NC2CCCC2)CCC(OC2CC(N3CCC3)C2)CC1 N1(C(CC(C)CNC(=O)CN2CCCC2=O)=O)CCC2(CC1)CC2CO c1(C(=O)NC2CC3(C(NC(C(C)CF)=O)C3)C2)cnc2c(c1)COCC2 C1(C(N(CCC)CCNC(c2ccon2)=O)=O)CC12CCC1(CC2)OCCO1 N1(C(CCCCN(C)C)=O)CCC(C2CC2)C1CNC(c1ccc(=O)n(O)c1)=O C1(NC(C(C)N(C)C)=O)CCN(C(=O)CCc2ncccn2)C(C)C1 c1(C(N2CCC(C3CCCN3C(c3cncnc3)=O)C2)=O)cc2cc(Cl)sc2[nH]1 N1(C(C2(C)C(C)C2)=O)CCC(CCNC(c2ncoc2Br)=O)C1 C1(C(C)(C)C)(CNC(c2c(C)scn2)=O)CCN(C(C2CCS2(=O)=O)=O)C1 c1(C(=O)NC(C(CO)NC(CCCOC(C)C)=O)C)cc2c(nn1)OCCS2 N1(C(C(C)=C(CC)C)=O)CCC(c2n[nH]cc2CNC(=O)CC2(O)CCC2)C1 CC1(C)CCC(C(=O)Nc2cc(C#N)ccc2F)CN1C(=O)C=Cc1nccs1 N1(C(C2C(CC)OCC2)=O)CC2(CCC(NC(=O)Cc3cnccc3Cl)CC2)C1 c1(C(C)C)n[nH]c(=NCC(C2CCCCC2)NC(C2CCS(=O)(=O)C(C)C2)=O)o1 N1(C(C2N=C(C)SC2)=O)CCC(C(C)NC(c2ccccc2OC(F)F)=O)CC1 C(=O)(C(F)CC(C)(C)NC(C1CN(C(N)=O)C1)=O)N(C)Cc1ccco1 C1(NC(CC(=C)C)=O)CS(=O)(=O)N(C)C12CCN(C(=O)C(O)CC(C)(C)C)CC2 C1(N(C(C2CCC(F)C2)=O)CC)CCC(NC(c2ccc(Cl)o2)=O)CC1 N1(C(C2N(C(C#CC(C)(C)O)=O)CCC2(C)C)=O)CC2CCCC1C2CO Cc1nn[nH]c1C(=O)NC1CC1NC(=O)Cn1cc(I)nn1 CCCC(CCO)CN=c1[nH]c(N2C3CCC2CC2(CC2)C3)nc(=NC)[nH]1 c1(C(N(C)CC2N(C(c3cc(CC)on3)=O)CCC2)=O)ccc(C)nn1 N1(C(CCC2OCC(C)(C)C2)=O)CCCC(CNC(c2occc2Cl)=O)CC1 c1(C(=O)NCC(C)NC(c2nnn(COCC)c2N)=O)ccc(S(C)(=O)=O)[nH]1 c1(C(c2cn(C(C)CNC(c3cnc(C)o3)=O)nn2)COC)ccc(F)cc1 c1(CC(=O)N(C(CNC(CC(C)N2CCCC2=O)=O)C)C)cc(F)cc(F)c1 CC1CC(NC(=O)C(C#N)CC2CC2)CCN1C(c1cc(F)c[nH]1)=O C1(CNC(=O)CC2CCOC2)CCCN(C(c2ccccc2C(F)F)=O)C1 c1(C(N2CCC(C)(CNC(COCCC)=O)C2)=O)cscc1S(C)(=O)=O CC1=C(C(=O)N2CC(CC(C)(C)CNC(c3ccco3)=O)C2)CCC(C)(C)C1 C(=O)(C(C(C)NC(C1CN(S(=O)(=O)c2cccnc2)C1)=O)C(C)C)OCC C1(NC(CCc2nc(C)c(C)[nH]2)=O)CCN(C(=O)CN(C)C(C)C)C(C)C1 C1(C2CN(C(C3COCCO3)=O)C2)(NC(CC(=O)OC)=O)CC1 C(=O)(C1=CCC(C)CC1)NC1C(C)CN(C(=O)CCSCc2ccccn2)CC1 c1(OC)cc(C(=O)NCC2(CCNC(c3csc4cncn34)=O)CC2)c(Cl)cn1 C(=O)(CC(O)CCc1ccccc1)NCC(CC)(CC)SC C=CCCC(CC(C)C)C(=O)NCc1nc(CNC(=O)C(CCC)OC)cs1 C#CCC(C)(C(=O)NCC(=O)N(C)O)N(C(=O)C(c1nocc1C)C)C.n12cc(nn1)[nH]c2=O.C CCCC(CC(=O)N1CC(C(C)OC)C1)NC(=O)CC1CCC(=O)C1C c1(CN2CC(F)CC(C(=O)Nc3c(C(N)=O)cc(C)s3)C2)cnc2[nH]ccc2c1 C1(C(=O)NC2CC2)CCCCC1C(=O)NCC(F)(F)C(F)F c1(CNC(C(C2CC2)OC)=O)cc(C(=O)NC2(C(N)=O)CCCCC2)ccn1 c1(C(=O)NC(CSCC)C(=O)NCC2CCC3CC23)csnc1Cl C1(NC(=NCCC)NCC2CCN(Cc3ccccc3)C2)CCC2(C1)OCCO2 C(CC(C)(C)C(=O)NOCCC(C)O)NC(C(C)OCCCC)=O C1(C(=O)Nc2c(C)cnc(Cl)c2)CCc2nc(C(F)(F)F)cn2C1 C1(C)(C(=O)Nc2scc(C)n2)CCCN(C(c2ccnnc2)=O)C1 c1(NC(C2CC2CNC(C(CCCOC)C)=O)=O)cc2oc(Cl)cc2[nH]1 C1(CNCc2nc(CCC(C)C)on2)CN(C(=O)OC(C)(C)C)CCN1C Cc1cc(CN2CC(O)(C(C(=O)NC(c3ccc(Cl)s3)(C)C)F)C2)on1 C=CCCC(C(=O)OC)NC(C1CN(C(=O)C(F)C(F)(F)F)CC(C)O1)=O C(c1ccc(F)cc1F)=CC(N1CCC(NC(=O)Cc2cnc[nH]2)C1C1CC1)=O N1(C(C(CC)O)=O)CC2(CCC2)CCC1CNC(=O)C(C)CC1CCC1 c1(C(=O)NC2CN(C(CCN(C)CC)=O)CC2N=[N+]=[N-])ccc(F)c2[nH]ccc12 c1(CN2CC(C)(C)N(CC(c3ccsc3)O)CC2)ccc2c(c1)CCC(=O)N2 N1(CC(=O)NCC2(NC(C(C=CC)O)=O)CCOC2)CCC(O)CC1 c1(C(C(=O)NC2C(CNC(C(C)(C)OCC)=O)CCC2)(F)F)ccc(Cl)cc1 N1(C(=O)OC(C)(C)C)CCc2ncc(C(=O)OCc3ncccc3F)n2CC1 c1(N2C(=O)CC(C(N(C)Cc3ncc(Cl)n3C)=O)C2)cc(F)ccc1F c1(N2CC3C(CNC(C4CCCO4)=O)C3C2)ncnc2sc3ccccc3c12 C(=O)(C(C(C)(C)C)N(C)C)NCCn1ccc(C(N(CC(O)COC)CC)=O)c1 CC1CN(C(c2cc(F)cnc2OCc2ccccc2)=O)CCC1N(C)C C1(NC(C2C(C)(C)CCO2)=O)CN(C(c2cnn(C3CCCC3)c2)=O)CC12CC2 C1(NC(C2C3CN(C(CC(C(C)C)C)=O)C2C3)=O)CCCCN(C)C1=O c1(CC)cc(CC(N2CCCC2C2(NC(c3cnc(C(=O)OC)s3)=O)CC2)=O)on1 C(C(=O)N1CCCC1C(C)NC(c1cccc(F)c1F)=O)(C(C)(C)C)OC c1(OCC)cc(C(N2CC3CN(C(=O)C4CC4)CC23)=O)ccc1OC C1(NC(CCc2onc(CCC)n2)=O)(CO)CCN(C(C2CCCN2C=O)=O)C1 C1(CCNC(C(CSC)C)=O)COCCN1C(c1cnc(C(F)(F)F)cn1)=O C1(CC(=O)NCC2CC(NC(CCN(C(CCC)C)C)=O)C2)CC(=O)NC1=O C1(CCC)CCCN(C(=O)NC2COCC2N2CCCCC2)C1 C1(C(=O)NCCC(C)C(F)F)CCN(C(C2C=CCS2)=O)C12CCC2 N1(C(CC=CC)=O)CCN(C(C2C3CC4C(C3=O)C24)=O)C2CC12 CCC(CC(=O)NCC1CCC(C(=O)N(C2CCC(C)(C)C2)C)C1)C(C)C CCCCC(CC(=O)NCc1cc(O)ccc1F)NC(C1SCC=C1C)=O C1(CNC(C(c2cn(CC)nc2)=O)=O)CCN(Cc2cnn[nH]2)CC1C CC(C(=O)NCCCCNC(=O)CCc1c(Cl)cccc1Cl)S(C)(=O)=O C1(CNC(C=CC=CCCCCC)=O)CC12CCN(C(C1CCC(=O)O1)=O)CC2 c1(C(=O)NCC(C)NC(=O)C(C(C)O)N(C)C)cc(F)ccc1F C(CC(C)NC(=O)C(c1ccoc1)NC(=O)COCCN(C)C)SCC c1(C(N(C2CN(C(c3c(C)cc[nH]c3=N)=O)CC2F)C)=O)ccc2cncn2c1 N1(C(C(COC)O)=O)CCC2(CCCCN(C(=O)Cc3ncc(C)s3)C2)C1 C1(NC(c2n(CC#C)ccc2)=O)CC2(CCN(C(=O)CCC)CC2)C1 C(c1cc2ccccc2o1)=CC(N1CCC(O)(CC(=O)NCC(=C)C)C1)=O C12(C(=O)NCC3C(NC(c4nc(Cl)cs4)=O)CC3)CC(C1)C(c1ccccc1)O2 C1(C(=O)NCCc2ccnc(C)n2)CCC2CCC1N2C(c1cn(C)cc1C)=O CC1CCN(C(=NCCc2cccs2)NCCc2ncc(Br)s2)C1 O=S(=O)(c1c[nH]ccc1=NCC(F)CO)NCC1(CO)CC=CC1 C(=O)(C#CC1(C)COC1)NCC1C(N(C(=O)C(C2CCCCC2)O)C)C1 c1(C(F)(F)F)cc(C(=O)O)ncc1F.c1(NCCOC)nc(CC)cs1 N1(C(CN(CC)CC2CC2)=O)CCC(NC(C2(CC3CCC3)CC2)=O)C1 N1(C(C(C)N(CC)CC)=O)CCCC2(CCN(C(=O)C(C(C)C)N(C)C)C2)C1 CCCC(C)(O)CC(=O)N(CCCNC(c1ccc(C(C)CC)cc1)=O)CC c1(CC(=O)NCC(CNC(C2C(C3C(C)C3)C2)=O)O)nc2ccccc2s1 C1(CNC(C2C(C(C)=O)C2(C)C)=O)C2CN(C(=O)CC3CCC(C)(C)O3)CC12 c1(CNC(C2(CC=C)CN(C(CCCC=C)=O)C2)=O)ccc(C)cc1C N1(CC=C)CCN(C(C23CC(CO2)N(C(=O)C(C)(C(=O)OC)OC)C3)=O)CC1C c1(C(=O)NC(CC(C)NC(=O)CC2CCCCC2O)C)cnc2nccnc2c1 C1(NC(C2C(OC)CCC2)=O)CCCN(C(=O)Cc2c(O)ncnc2O)CC1 Cc1cc(F)c(C(=O)NCC(C)CN(C)C(C23CC(C2)S(=O)(=O)C3)=O)c(F)c1 c1(C(=O)NC2CN(Cc3cc(OCC)cc(F)c3)CC2F)cc(Br)cc(F)c1C C12CCCN1C(=O)C21CC1.C(C(=O)NCCCNC(=O)CC)=CCC C1(C2(NC(c3c(C)con3)=O)CC2)CCCCN1C(c1cccc[n+]1[O-])=O N1(C(CC(C(C)C)C)=O)Cc2ccccc2C(NC(c2c[nH]nc2C2CC2)=O)C1 C1(N(C(C2CCC(F)C2)=O)CC2CCCCO2)CCC2(CC1)CNC2 c1(C(N2CCCC(CC(=O)NCCCOC=C)CC2)=O)c(Cl)ccc(F)c1Cl Cc1cc(C(N2CC(F)(F)CC2CNC(C2CCC(F)C2)=O)=O)n2ncnc2n1 C1(COC)(NC(=O)Cc2ccnn2C)CCN(C(=O)Cc2c[nH]nc2C)CC1 Cc1nc(C=CC(N2CCC(NC(=O)CCCC(N)=O)C(F)C2)=O)[nH]c1C C(C(=O)NCC(C(=O)NCC1CCCCO1)N(C)C)(C(C)(C)C)N(C)C C(CCC(N)=O)(C(=O)N1CCC(NC(=O)OC)C1)n1cc(CN(CC)CC)nn1 CC(C)CC(O)CC(=O)N1CCCC(C)(CNC(=O)CC2CCOC2)C1 CC(C)CCCCN(C)C(c1c(CNC(c2cc(O)ncn2)=O)nnn1C)=O C1(C(N(CCCN(C)C(C2CCCC3CC23)=O)C)=O)CC2CCC1CC2 Cn1cc(C(=O)NCC2CCN(C(=O)C(F)C3CCC3)C2)c2ccccc2c1=O n1(CC(N2C(C)CN(C(C3CC3C(F)F)=O)CCC2)=O)cnc2c(N)ncnc12 C(=O)(CCCCC(F)F)NC(CC)(CNC(=O)CC1CCC(C(F)(F)F)O1)CC c1(CC(=O)NCCC2CC(NC(C3CC(=C)C3)=O)C2)cnn(C(C)C)c1 c1(C(C)NC(c2n(C(CC)C)ncc2)=O)cnccc1OC c1(CC(=O)NC(CC=C)CNC(=O)C(C)(F)F)cnc2n1CCCC2C C(C)(CC(=O)NC1(C)CN(C(C2(N3CCOCC3)CC2)=O)C1)(C(F)(F)F)N(C)C C1(CC)CCc2sc(C(=O)N(C3CCCN(C(=O)C(C)(C)CSC)C3)C)cc2C1 C1(CC(=O)NC2CN(C(C34CCCC3CCC4)=O)C2)CCS(=O)(=O)CC1 N1(C(=O)NC(c2c(OC)cccc2)CC)CC(=O)NC2CCCCC12 C1(NC(C2CC(=O)NC2)=O)CC2(C(=O)NC3CC(CO)C34CCC4)COC1C2 c1(CC)ccc(C(=O)NC2(CNC(=O)C(C)Oc3cccnc3)CCOC2)cc1 c1(C(N(CCCCN(C(c2c(SC)cccc2)=O)C)C)=O)noc2c1COCC2 C1(NC(Cc2nc(C)sc2)=O)CN(C(C2CCCSC2)=O)CC1n1cccn1 C1(NC(C2CCN(CC(C)C)C2)=O)C2CN(C(C3CSCCS3)=O)CC12 C1(NC(CC(=O)NCC)=O)CCN(C(c2cnn(C)c2C2CC2)=O)CC1C C(C)(C)(C(=O)NCC1CCN1C(c1ccc(C(C)=O)[nH]1)=O)OCC C(=O)(C(C)(C)C(F)F)NC(C1(O)CN(C(c2c(C)[nH]cc2)=O)C1)C Cc1cc(C(N2CC(NC(c3cccn3C)=O)C(F)C2)=O)cc(Cl)c1Br c1(C(=O)NCC2CC(CNC(CCSC)=O)C2)cn(C2CCOC2)nc1C C(=O)(C(CC)C(C)(C)CC)NC1(C)CN(C(c2cccc(CC)n2)=O)C1 O=C(C1CCCc2ncccc21)NCCC1(NC(=O)C(C2CCOCC2)O)CC1 N1(C(CCc2c(C)ncs2)=O)CCCC2CCN(C(=O)C3=CCSC3)CC12 C1(NC(c2cnc(CCC)s2)=O)CCN(CC(N2CCNCC2)(C)C)CC1 c1(N(C)C)nc2cc(C(=O)NC3CCCC34CCCC4)ccc2o1 C(=O)(C1CCCc2sccc21)NCC(C)CN(C)C(C1(C(F)(F)F)CCC1)=O Cc1cc(Cl)ccc1NC(C1CC12CCN(C(=O)CCNC(N)=O)C2)=O c1(NC(C(C)CN(C(=O)C(F)CC2CCOC2)C)=O)ccc(O)c(=O)cc1 N1(C(C=C(C)C)=O)CC2(C(=O)NCC(C)(O)C3CCC3)CCC1CC2 C(C)(C(C)C(=O)NCC1(CC)CCOCC1)NC(C1(CC)CC1)=O Cc1[nH]c(C#N)cc1C(=O)NC1CC(O)CN(C(=O)C(C)(C)C(C)C)C1 C(=O)(CC(C)P(C)(C)=O)N1CCC(C(N2C(CCC(C)C)CCC2)=O)CC1 C1(NC(C(CC)n2cccn2)=O)CN(C(c2cc(Cl)n[nH]2)=O)CCC1O c1(C(N2CCN(C(C(C(C)C)OCC)=O)CC(C)C2)=O)c[nH]c2nccc-2c1C C#CCCCC(C)(c1nnnn1-c1ccc(F)cc1)NCC(CC)CCCC Cc1nc2ccccc2c(C)c1C(=O)NCCNC(C1CC(C)(O)C1)=O Cc1nn[nH]c1C(=O)NCCC(C)NC(c1cc(Cn2cccn2)on1)=O C1(NC(C2C(CNC(C=CCOCCOC)=O)CC2)=O)CCCC1C n1(CCC(=O)NC2C(CNC(=O)CSCc3ccncc3)C2)cc([N+](=O)[O-])cn1 C1(C(=O)NCC2N(C(c3c(CC)cco3)=O)CC(O)C2)CC2C(C1)C2(F)F CCC(CC(=O)NCC(CCNC(C1CC(O)CN1C)=O)OC)C1CC1 C=CC(C)(O)CC(=O)N1CCCC1COCC.NCC CCCCC(CC(=O)NC1COCC1NC(N)=O)NC(C1CC2(CCC2)C1)=O Cc1ccc(C(N2CC(NC(C3CCC(=O)N3)=O)C2)=O)nc1C c1(OC)cc2cc(c1)C(c1cccc(Cl)n1)N2.c1(CC(=O)OC)nn[nH]n1 C1(NC(C2CCC(NC(C(C)OCCOCC)=O)CC2)=O)CCC2(CCC2)CC1 C(=O)(CCCCCOC)NC1C2(CC(NC(C3N(C(CC)=O)CCCC3)=O)C2)C1 Cc1cc(C(=O)NC(c2cnn(C)c2)C(=O)N(C2CCCC(C)C2)C)[nH]c1C N#CC1(c2ccccc2)CC1C1CCCN1n1cc(CCS(C)(=O)=O)nn1 c1(C(N2CCC(C)(COC)C2)C(=O)NCCCCCC)ccc(F)c2[nH]ncc12 CCCCCCCCCCC(=O)OCN1CCCC1C C1(C(N2CCC(CN(C(C(CC#C)C)=O)C)C2)=O)Cc2ccccc2CO1 c1(NCC2(CC)CC2)nc(=NC2CCN(CCF)C2)[nH]c2c(C)nn(C)c12 CCCC(CCCNC(c1ccc(F)s1)=O)NC(=O)C(C)(C)COC C1(C(=O)NC(CN(C(CC2N(C(C)C)CCC2)=O)C)C)CCc2nncn2CC1 C#Cc1cc(C(N2CCCC(F)(C(N3CCCC3CC(N)=O)=O)C2)=O)ccc1C Cc1nn(C)cc1NC1(c2nnnn2C2CCCC2)CCC1CC(F)(F)F c1(C(N2CC3(N(C(Cc4cccc(C)c4)=O)CC3)C2)=O)cnc2c(cnn2C)c1 c1(OC)c(Cl)nc[nH]c1=NCC1(O)CN(C(=O)C(C)(C)n2cnc(C)c2)C1 N1(C(c2c(C)noc2C)=O)CCN(C(=O)CSc2ccncc2)CC(C)(F)C1 c1(OC)cc(CN2CCNCC2C(=O)Nc2ccc(Cl)c(I)c2)cc(F)c1O C1(CNC(c2ccc(OC(F)F)nn2)=O)COCCN1C(=O)CCC1CC1(F)F N1(C(c2c(N)cc(Cl)nc2)=O)CC2CCC(NC(C3CSCC(=O)N3)=O)CC2C1 C1(C(=O)NCCC2CCN(C(c3c(COC)cco3)=O)CC2)CN(C)CC(C)O1 Cc1cc(O)ncc1C(N1CC(NC(=O)CCc2cccc(Cl)c2)C(O)C1)=O CCCCC(CC(=O)NCCC1CC(=O)N(C)C1)NC(=O)C(C)(C)NC(=O)OC N1(C(Cc2cc(CC)no2)=O)CCCC(F)(CNC(=O)Cc2cccnc2Cl)C1 N(C(=NCCN(c1ccccc1)C(C)C)NCC1CCC(F)(F)CC1)C(C#C)C C(C(C)(C)C(=O)NC(c1nn[nH]n1)CC)NC(CC=C)=O C1(NC(N(c2c(C)nsc2)C)=O)CCCC(OC(F)F)C1 C1(C(N2CCC(NC(C(CC)=CCCC)=O)CC2)=O)CC2(CCC2)CO1 c1(C2(C(=O)NCCC(O)CNC(C3CC3(F)F)=O)CCCC2)cccc(Cl)c1 CC1(C)CCCC(OC(=O)Cn2ccc(C(F)(F)F)n2)C1 C(=O)(C(C)CC(C)(F)F)N(C1CCN(C(c2c(C)ccnc2C)=O)CC1)CC Cc1cc(C(C)C(=O)NC2CCN(C(=O)C=CC(=O)N(C)C)C(C)C2)cc(C)c1 c1(C(=O)NC2(CO)CCC(CC)CC2)cc2sc(C)c(C(=O)O)c2[nH]1 c1(C(=O)NCCCCCNC(c2ccc(O)cc2)=O)ccnc2ccsc12 C12(C(N(C(C(=O)NC3(C(=O)OC)CCC3)C)C)=O)CSCC1C2 CCCCCCC(c1nnnn1CCCOCC1CC1)NC1CC(F)C1 Cc1ccc2[nH]nc(C(=O)NC3CCCC3NC(c3cc(Cl)ccc3C)=O)c2c1 C1(CNC(C23CC(C(C)C)(C2)C3)=O)N(C(c2ccc(O)cc2)=O)CCCC1(C)C Cc1ccc(Br)cc1NC(=O)NC1COCCC1OC(F)F C1(NC(CCC(=O)N(C(C)C)C)=O)CN(C(c2occc2C2CC2)=O)CC1(C)C C1(CNC(c2cnn(CC)c2C)=O)CCN(C(=O)CC(C)C2CCCC2)C1(C)C C(=O)(C(C)C(O)C(C)C)N1CC=C(C(=O)NCC(CC)CC)C1 CN1CC=C(CNC(=O)CC2CCCC2NC(C2C3CCC(F)C23)=O)CC1 C1(CNC(C(C)OCCC(C)C)=O)CCCC1NC(c1ccsc1C(F)F)=O C1(O)(Cn2cc(CCN(C)CC)nn2)CCCN(C(=O)C(F)CC(C)(C)C)CC1 Cc1cc(F)c(N)cc1C(=O)N(C)CC1CCCC1NC(c1ccccc1)=O N1(C(CC(=O)NCC)=O)CCOC(CCNC(=O)CCOCC2CC2)C1 CN1CC2CC1CN2C(=O)CC1CN(C(=O)CCc2ccccc2)C(C)(C)C1 c1(CC)cc(C(=O)N(CCNC(c2cccc(SC)c2)=O)C2CC2)nn1C c1(CC(N2CC(CC(C)NC(CCOCC)=O)C2)=O)cc(C2CC2)no1 N1(C(C(CC)NC(C)=O)=O)CCN(Cc2ccccc2)C2CC12.OC C(=O)(C#Cc1ccnn1C)N1C(N(C(c2ccc(NC)cc2)=O)C(C)C)CCC1 N1(C(C(=O)N(C)C)=O)CC2C(NCCCc3nnsc3Cl)C2C1 N1(C(C(F)=C(C)C)=O)CCC(NC(=O)CC2CCC(=O)N2C)C2(CCC2)C1 c1(C(=O)OC)cc2c(cc1F)CCN(C(=O)NC1CCC3(CCC3)OC1)C2 N1(C(Cc2c(C)nn(C)c2)=O)CCCC(CNC(=O)C(C)(C)n2ccnn2)CC1 N1(C(c2sc(C)c(O)n2)=O)CCCC(C2CC2NC(=O)Cc2ccnc(F)c2)C1 N1(C(CC2ON=C(CC)C2)=O)CCC(C)N(C(C2CN(C(N)=O)C2)=O)CC1 c1(N2CCC(N(C(=O)Cc3cnnn3C)CC)C2)ncnc2sc([N+](=O)[O-])cc12 C1(C(=O)NC(c2ccsc2)C)CCC(NC(=O)Cc2cscn2)CC1 C1(C2CC2)(CNC(c2c(CC)noc2)=O)CCN(C(=O)CC(=O)NC2CC2)C1 c1(C(=O)NCC2C(C)CN(C(c3ccnn3C3CC3)=O)C2)cncn(C)c1=O CC(C)CC(=O)C(=O)NC1CC(CCC(N2CCCC2C(C)(C)C)=O)C1 C1(OCC(=O)NCCNC(=O)C(CO)c2ccccc2)CCCCC1 c1(OCC)cnc(C(=O)N(C2CCCS2(=O)=O)c2ccccc2)cn1 C1(C(N2C(C(=O)Nc3c(C(=O)OC)sc(C)c3)CC2)=O)CC(C)(C)CC(C)(C)C1 CC(C)(CC(=O)N1CCC1CC(=O)NC1CCC(O)C1)n1cccc1 C1(C(=O)NC(CC(C)NC(=O)CN(CC(C)(C)C)C)C)CCc2nc(O)[nH]c2C1 C(=O)(C1=CC(C)CC1)N1CCC(CC=C)(NC(=O)C=COCC)C1 C(=O)(C(C(=O)N1CCC(CNC(=O)C(c2cnn(C)c2)O)CC1)OC)OC C1(C(=O)NCC(C2CCCCC2)O)(CC)CCN(C(=O)CCC2CC2)C1 C(=O)(C=CS(C)=O)NCC(n1cc(NC(=O)CSCC(N2CCCC2)=O)nn1)C C1(C(=O)NCCC(=O)OCC)CCN(C(C23CC(C)(CCO2)C3)=O)C12CCC2 C1(C(=O)OC)CCC2(CCCCC2)N(C(C2CCOCC2)C(=O)NCCC#N)C1 c1(CNCC#CC)cn(C(C)C(=O)OC)cn1 Cn1nc(C(N2CCC(NC(C3COCCOC3)=O)C2C2CC2)=O)cc1Cl c1(CNC(C(C2(C)CC2)NC(CCN(C)CC)=O)=O)nn[nH]c1C1CC1 CC(C)(CC(F)C(=O)NC1(CC2CCC2)CC1)NC(=O)C(F)C(F)(F)F CC(CC(=O)NCC(C)NC(=O)C=Cc1ccccc1Br)CC(F)(F)F S(=O)(=O)(c1cccc(=NC(C)CC)[nH]1)N(CC)CC.C1CC(C)N1 CC1CC(C)N(C(=O)COc2cn[nH]c2)CCN1C(c1cncc(C2CC2)c1)=O N1(C(CN(C(C=NOC)=O)C)=O)CC(SCC(=O)OC)CC(C)C1 c1(C(N2CCC(C(C)NC(=O)COC3CCCOC3)CC2)=O)cc(O)nc(O)n1 Cc1c(C(N2CCCC(C(C)C(=O)NC3(C(C)C)CCC3)C2)=O)cnn1C CCS(=O)(=O)c1ccc(Cl)c(C(=O)NC2C3CC2N(C(=O)C2=CCOC2)C3)c1Cl N1(C(C(CC=C)C)=O)CCN(C(c2cccc(Br)c2)=O)CC1CC1CC1 N1(C(c2cc(CNC(C3(CC)COC3)=O)nn2C)=O)CC(F)(F)C(F)(F)C1 N1(C2(C3(NC)CCC3)CC2)CC2(CC(C(=O)NS(C)(=O)=O)CO2)C1 O=C1CCC(C(=O)NCC2CC2CNC(=O)CN2CC3CC3C2)=NN1 C12(NC(Cn3ncc(C#C)c3)=O)CCOCC1CN(C(c1cc(=O)cc[nH]1)=O)C2 CC1(CNC(c2c[nH]nc2F)=O)CCC(NC(C2CC(CC(F)(F)F)C2)=O)CC1 c1(C(=O)NCC2CCN(C(C3(SC)CCC3)=O)C2)cc(C)c2c(c1)CCC2 N1(C(C(N2CCOCC2)C)=O)CCCCC1C1(NC(=O)C=CCF)CC1 C1(C(=O)NCC(C)N(C(=O)C(F)=C(C)C)CC)CCOC1c1nccn1C C1(C)(NC(COCCC)=O)CCCN(C(c2ccn(C)c2C)=O)C1 CC(=O)CCCCC(=O)N1CC(O)(C(F)C(=O)NC(C)(C)C(C)(C)O)C1 C1(C(=O)NC2(C)CCCS2(=O)=O)(C(=O)O)Cc2ccccc2C1 N1(C(C2(CC)CCOCC2)=O)CC(CNC(=O)C(C)C(C)(C)C)CC(C)C1 c1(C(C(=O)N(C(C)CNC(=O)C(C)(C)NS(C)(=O)=O)C)=O)cccc(Cl)c1 C12(CC(=O)NCN)CCC1CN(C(=O)CN1CCOCC1=O)C2 c1(C(N2CCC3(CN(C(C4CC(C)OCC4)=O)C3)C2)=O)cc2c(cc1Cl)NCC2 C12(CNC(CC3CC(=C)C3)=O)CC(NC(=O)C(=O)NCCOC)(CO1)C2 CS(=O)(=O)c1cccc(NC(C2CCN(c3ncnc4n[nH]cc34)C2)=O)n1 c1(C(C)C)ccccc1C(N1CC(CN(C(=O)CC(C)C2CC2)C)C1)=O c1(C(=O)NCC2(NC(CN(C3CCCC3)C)=O)CCOC2)ccc(Cl)cc1N N1(C(C(C)SCCCC)=O)CCC2(CCN(C(=O)CC(=O)OC)C2)C1 c1(OC)ccc(OC)c([N+](=O)[O-])c1C(N1CC(N(C(=O)C2=CC(C)(C)C2)C)C1)=O c1(SC)cscc1C(=O)NCC1(CNC(C2CCCN2C)=O)CCC1 C1(C2CC2)(CNC(C(CCC)(C)O)=O)CCN(C(=O)C=C(Cl)Cl)C1 N1(C(COCCSC)=O)C(C(=O)N(C)Cc2cncn2C)CC2CCCC12 c1(C(=O)NC2CN(C(Cc3ncc(C)o3)=O)C(CO)C2)c(C)ccc2n[nH]cc12 c1(NC(N(C(CC)C)C)=O)ccc(C(F)(F)F)cc1C#N c1(C(N2CCC(NC(C(CCC)N(C)C)=O)C23CC3)=O)ccc(C#N)c(C)n1 c1(C(C2CCOC2)C)cn(CC(F)CCNC(=O)C(c2ccccc2)C)nn1 C#Cc1ccc(CNC2(c3ccc(-c4cccc(C5CC5)c4)nc3)CC2)cc1 C1(C2CC2)(CNC(CC2(C)CC2)=O)CCN(c2ncncc2Br)C1 C1(CC)CCC(C(N2CCC(N(CCO)C(c3coc(N(C)C)n3)=O)C2)=O)O1 c1(SC)ccccc1C(=O)NCC(c1ccccc1F)NC(=O)C=CS(C)=O C1(N(C(C2C(=C)C2)=O)C)CN(C(c2csnn2)=O)CCC1O N1(C(Cc2cc(C)no2)=O)CC=CCC1C(=O)N(C1CC(O)C1)C N1(C(C2C(C(C)NC(CN(C(C)=O)C)=O)C2)=O)CCC2(CNC(=O)O2)C1 c1(C(=O)NCC2CCN(C(c3nnn(C(C)(C)C)n3)=O)C2)ccc2c(n1)NCC2 C1(C(=O)NCCC2CN(C(C(CC=CCC)C)=O)C2)Cc2nnc(C)n2C1 C1(F)(C(=O)NC2CC(C(=O)NCCC(=O)NC(CC)C)C2)CCOC1 C(CCC(C)(C)NC(=O)C(F)n1cccn1)NC(C(CSC)O)=O C=CCCCC(C)(C)CNC(=O)C(C1CC1)N(C)C(C1CC2CC1CC2=O)=O C1(CN(C)C(C2(C)CSC2)=O)CCCC(NC(=O)C=CBr)C1 N1(C(C2(CC)CCCN(C(c3ccc(O)cn3)=O)C2)=O)CCCC2(CC(O)C2)C1 c1(C(=O)NC(CCNC(C2C(C(=O)OCC)C2)=O)C)ccncc1-c1ccccc1 C(c1cnn(C)c1)=CC(=O)N(C)CC1(CNC(C(N2CC(C)C2)C)=O)CC1 CCCCC(CCC)CN=c1[nH]c(=NCCN2CCOC2=O)[nH]c2ccsc12 C1(CCCC)CN(C(=O)CC2CCC2(F)F)CCN1C(=O)CSS(C)(=O)=O C1(NC(c2cc(CCC)on2)=O)CC2CCC1CC2NC(=O)CN1CCC(C)C1 c1(COC(N(CC(CC)(F)F)Cc2ccccc2)=O)ccc(N)cc1I c1(C(CC)=O)ccc(NC(C)(C(C)C)c2nnnn2C(C)CC)cc1 C1(CCC(=O)NCCCN(C(=O)C(CC2CC2)CC2CC2)C)CCC(=O)NC1 C1(C(=O)OC)CCC(c2cnc[nH]2)N1C(=O)C(C)Cc1c(C)noc1C N1(C(C(CC=C)NC(=O)Cc2ccc(C#N)cc2)=O)CCc2cncnc2C1 N1(CC(=O)NC2CC3(CC(NC(C(C)=CC)=O)C3)C2)C(=O)c2ccccc2C1=O C1(C(C)C)COCCN1C(C1CCCCC1NC(C1CC1CCN(C)C)=O)=O c1(-c2nc(SCc3c(N(C)C)ccc(Cl)c3)nn2C)cccc2nncn12 n1(NC(=O)C=CC(=O)OC)nc(C)c2cc(C(=O)NC(CCCCOCC)C)sc12 C(=O)(C1=CC2(CCOC2)C1)N1CC(OC)C1.C(=O)(CCNC1CCCC1)C(=O)CO CCC(CC(=O)N1CCC(N(CCO)C(C2CCCO2)=O)CC1)C(C)C c1(CC(N2CCC(NC(C3CCC(CC)O3)=O)C2)=O)sc(C)nc1C N1(C(C2(O)CC2)=O)CCC2CN(C(=O)C(F)(F)c3cnc(C(F)(F)F)s3)CC12 Cc1nc(C(=O)N(C2CCN(C(=O)CP(C)(C)=O)CC2)CCCO)cn(C)c1=O C1(CNC(=O)CC(O)C2CC2)CCN(C(=O)C=Cc2ccccc2)CCC1(F)F C1(C)(C(=O)NC(C=CC(=O)N(c2cnn(C)c2)CC)C)CC2CC2C1 Cc1c(C(=O)NC2CC(NC(C3CC4CCC(C3)O4)=O)C2)cc(O)cc1N CC(C)CCC(O)C(=O)N1CC=CC1(C)C(=O)NC1CCn2cnnc2C1 C1(C(=O)NCc2cn(C3CCN(C(CCOC(C)=O)=O)C3)nn2)CCCC1(F)F C(CC(F)F)(C(=O)NOCCCF)NC(C1CCCCO1)=O N#Cc1n[nH]c(=NC2CC(O)(CNC(c3c[nH]c4ccccc34)=O)C2)s1 N1(C(c2cc(C)ncc2)=O)CC2(CNC(c3cnc(N(C)C)nc3)=O)CC1CO2 n1(CC(=O)NCC2(COC)CCCN2C(C2CCC(O)C2)=O)nc(Cl)ccc1=O N1(C(C2C(=C)CC2)=O)CC2CCN(C(c3cccc(N(C)C)n3)=O)C2C1 Cc1ncoc1CN(C(=O)C(=O)N(CCc1ccccc1)CC1C(N)C1(C)C)C C1(NC(c2c(C(C)C)nns2)=O)CCCC(NC(c2cc3ccsc3s2)=O)CC1 N1(C(C(C(CC)(C)C)=O)=O)CCC(C(=O)NCC(C)C(C)C)=C(F)C1 c1(C(N(CCNC(c2cc(C)c(C)o2)=O)CC)=O)csc2cccnc12 Cc1nn(C2CC2)cc1C(N1CCC2CC12C)C(=O)NC1CCOC1 C#CCC(CC#C)C(=O)N(CC(CO)(CO)NC(=O)CCc1ccncc1)C c1(C(N2CC(C=C)C(NC(=O)C(C)NC(N)=O)C2)=O)cc2c(F)cc(Cl)cc2[nH]1 N1(C(C#C)=O)CCc2c(C(=O)O)cccc2C1.N12CCOC(C1)C2 c1(CNC(CN2C(Cc3n(C)cnn3)COCC2)=O)cc2nc(F)ccc2o1 c1(C(=O)NCC2CN(C(c3c(C#C)cn(C)n3)=O)CC2C)cc2cc[nH]c2cn1 c1(C(N2CCCC(N(C(=O)C=CC(C)C)CC)C2)=O)ccc2nn[nH]c2n1 S(=O)(=O)(c1ccc(Cl)nc1)NC1CC2(CN(C(=O)C3=CCCC3)C2)C1 CC#CCCCC(=O)NC1CN(C(C2CNC(=O)N2)=O)CC1(C)C C1(C)(C(N(CC(C(=O)N2CC(C(C)OC)C2)C)C)=O)CCCN1C C1(NC(=O)C=CCO)CC2CC1CN(C(c1cnccc1C(F)F)=O)C2 c1(C(N2CC(NC(C3C(C)=C3)=O)C(C)C2)=O)cc(C#N)ccc1O C1(NC(C2(C(C)C)CCN(C(=O)C=Cc3cccnc3)C2)=O)CCCC(C)(C)C1 c1(NC(=O)NC(c2ncc(C3CC3)o2)(C)C)cc(C(F)(F)F)ccc1O c1(C(=O)NC(CN(C(COCC=C)=O)C)CC)nc(OC(C)C)ccc1Cl N1(C(CCCCCC)=O)CC(C)N(C(=O)C(F)C(CC)CC)CC1C C(=O)(C(=O)C(C)(C)C)NC1CC(C(=O)NCC(C#C)OC)CC1O C1(N(C(c2cccc(CC)n2)=O)C)CC2CCC(C1)N2C(=O)C(F)=C(C)C1CC1 C1(C2CN(C(c3cccc(CCO)c3)=O)C2)(NC(c2ncc(F)cc2F)=O)CC1 Cc1ccc(Cl)cc1OCC(N1CCC(NC(=O)C#CC(=O)N(C)C)CC1)=O c1(OC)nc(Cl)ccc1C(N1CCC(N(C(=O)CN2CCNC(=O)C2)CC)C1)=O C1(C(=O)NCCNC(C(C)NC(c2ccco2)=O)=O)CCCC1(F)F c1(CNC(C(CC2CCC2)NC(COCCOC)=O)=O)c(O)cccc1F N1(C(C(C)OC(=O)CCc2nccs2)=O)CCN(S(C)(=O)=O)CC1 C1C(O)CC(=O)N1.C(CCOCCN(C)C)NC(C1CSC1)=O Cc1nc(C(N2CC(NC(C3(Cl)CC3(F)F)=O)C(CC(C)(C)C)C2)=O)nn1C CCC(C)(C)C(C)CC(=O)NC1C(C)(C)C(NC(=O)Cn2nnnc2C)C1(C)C c1(C(N2CC(NC(c3cc(C)[nH]n3)=O)C(C)C2)=O)c(C(C)C)nn(C)c1Cl C1(CNC(C(C)CN(C)C)=O)CCCCCN1C(c1cc(=O)c(Br)c[nH]1)=O C1(NC(c2nc(COC)sc2)=O)CC2CC1CN(C(=O)CCCCCN(C)C)C2 N1(C(c2ncn(C(C)C)n2)=O)CCC(C)C(CNC(c2cc(Cl)c[nH]2)=O)C1 C=CCC(CC(C)C)C(=O)NCCC1(NC(=O)CCc2ccc(C)s2)CC1 c1(C(N2CCCC(NC(CCOC)=O)C(F)C2)=O)ccnc(P(C)(C)=O)c1 N1(C(Cc2c(C)nn(C)c2)=O)CCCCC(C(=O)NC(c2ccccc2)C)C1 C1(NC(c2c(SCC)cncc2)=O)CCN(C(=O)C=CCN(C)C)CC1O C1(CC(C)NC(C(C)=CC)=O)CC2CCC(C1)N2C(C1CC(C)CC(C)C1)=O CCC(CCOC)C(=O)NCC(CCOC)NC(=O)C(C1(O)CCCCC1)(F)F Cc1cn(C)nc1C(=O)NC1CC1NC(C1C=CCC1)=O C12(C(N(C(CNC(c3c(Cl)cn(CCC)n3)=O)C3CC3)C)=O)CCCN1CCC2 N1(CC(N2CC(OCCNC(Cc3c(C)n[nH]c3)=O)C2)=O)CCC(C)CC1 C1(CNC(c2ccc(CSCC)cc2)=O)CN(C(=O)CNC=O)CC12CCC2 C12(NC(=O)CC3CSCCS3)CCCN(C(c3nc(Cl)cs3)=O)CC1C2 N1(C(c2c(N)ccc(C)c2)=O)CC2CCC1C(NC(c1nc(Cl)c(Cl)s1)=O)C2 c1(C(=O)NCC(C(C)C(C)C)NC(C=CC)=O)oc2ccc(C)cc2c1C c1(OC)ccc(CCC(=O)NCC2CCN2C(=O)C(C)c2ccsc2)cc1F C1(NC(c2c[nH]cc2-c2ccccc2)=O)CCC(NC(C2OCCO2)=O)C1 N1(C(C(CCOCC)NC(c2ccc(C)nn2)=O)=O)C2CCC1CC1(CC1)C2 N1(C(CSCCC(C)C)=O)CCN(C(=O)CCc2ccc(Cl)c(F)c2)CC1C CC(C)C(O)CC(=O)NC(Cc1cnc[nH]1)C(=O)N(C1CCCC(O)C1)C C(=O)(C(C)(C)C(C)(C)O)N1CCC(N(C(c2cc(Cl)cnc2OC)=O)CC)C1 C(=O)(C(O)C(CCC)NC(=O)CCN(C)CCC)NC1(C#C)CCCCC1 C(CC(O)CC(=O)NCCCN(C(C1CC12CCOCC2)=O)C1CC1)SC c1(C(N2CC(NC(C(C)(C)OC)=O)C(C)C2)=O)cc(Cl)c(Br)cc1F C(c1ccc(CC)cc1)=CC(=O)NCC(CCNC(C(C)SCCCC)=O)(C)C C(CC(C)(C)CNC(=O)CC(C(F)F)c1ccccc1F)(OC)OC C(C(CC(F)(F)F)NC(=O)Cc1cscn1)NC(Cc1c(SC)cccc1)=O C(=O)(CC(=O)NC(C)(CNC(c1nc(-c2cnccn2)no1)=O)C1CC1)NC C(=O)(C1=COCCC1)NC(C1CCCCC1)CNC(C=C(CC)C)=O c1(C2C(C(=O)NCC(CNC(CCc3c(C)ncs3)=O)F)C2)ccc(F)cc1 C1(C(=O)NCCC(C)NC(C2(CCOC)CC2)=O)CCCCC1c1nc[nH]n1 c1(C(=O)NC(C)C(C2CCCCC2)NC(=O)C2=CCSC2)c(C#N)ncn1C C1(C(N2C(C(=O)NCCCCCC=C)CSC2)=O)CCOCC1(C)C c1(SC)ccccc1CNC(C1CC1NC(=O)Cc1ccnn1C)=O N1(C(C(Cc2cnc[nH]2)NC(C(CC)C#N)=O)=O)CCCN(C(=O)OC)CC1 c1(C(C(=O)NCC2CC(NC(=O)C(F)=CCCF)C2)=O)ccc(F)c(F)c1 N1(C(COCCCC#C)=O)CCC(C)C(NC(=O)C(C)CC=CCC)C1C N1(C(C2CN(C)C2)=O)CC2(NC(C3COC(=O)N3)=O)CCCC2(F)C1 Cc1cncc2cc(C(=O)NC(C)C(CO)NC(=O)C(O)c3ccsc3)sc12 c1(N2CCN(C(C34CCC(OC)(CC3)CC4)=O)CC2)ncnc2cccc(F)c12 C12(NC(C(C)OCC=C)=O)CCCC1CN(C(c1cccc3nnn(C)c13)=O)C2 C1(CNC(=O)C=CCN2CCCC2)CCC2(CN(Cc3ncc(Cl)s3)C2)O1 c1(CC(C(=O)NCCC2N(C(CCSC)=O)CCCC2)F)ccc([N+](=O)[O-])cc1 CC1(C(=O)NC2CCC(CNC(=O)CNC(c3ccsc3)=O)C2)C=CCCC1 c1(OC)cc(C(=O)NC2CCCC2NC(=O)C(C)CC(F)F)cc(F)n1 c1(C(N2C(CNC(c3cncc(C)c3C)=O)CC2)=O)cc2cnccc2[nH]1 c1(CC)nc(C(C)NC(=O)NCCc2cn(CCOC)nn2)cs1 N1(C(CCC(N)=O)=O)C2CCC1C(C(=O)NC1C3CC4C(C3)C14)C2 C1(CC(=O)N(CCNC(=O)CCOc2ccccc2)C2CC2)CC2CCC1O2 c1(NC(=O)NCc2cn(C3CN(Cc4onc(C)n4)C3)nn2)cccc(O)c1Cl C(=O)(C(C)CC(C)(F)F)N1CC(CNC(c2ccc(C)n2C)=O)OCC1 CC1(CNC(C2CC=CCO2)=O)CCN(C(=O)C(F)CC2CCOC2)C1 c1(C(N(c2cc(OC(C)C)ncn2)C2CCCNC2)=O)cccc(O)c1[N+](=O)[O-] Cc1cccc(CN2CC3C(NC(c4ccc(=O)n(C(C)C)c4)=O)C3C2)c1Br C1(NC(N2CCC(c3cnn[nH]3)C2)=O)C2Cc3ccccc3C12 C(=O)(C(CC)CCOC)N1CCC(N(CCC)C(C2C3CCCCC23)=O)CC1 CC1CC(NC(c2csc(C#N)c2)=O)CCN1C(c1cc(Cl)cc(Cl)n1)=O c1(OC)ccc(C(CF)NC(c2ccc(C(F)(F)F)cc2)C)cc1 C1(C(=O)NCC2(O)CN(C(C=Cc3c(C)cncc3)=O)C2)CC2(COC(=O)N2)C1 N1(C(c2ccc(C#N)s2)=O)CCC(F)CC1C(N1CCC(O)(CO)C1)=O C(=O)(CCCC(=O)N1CCN(C(=O)CC2CCC2)CC1)N(NCC)CC C(c1ccnc2ccccc12)=CC(=O)NCC1N(C(C(C(C)(C)O)F)=O)CCC1 N1(C(=O)C=Cc2ccoc2)CCC(O)(CNC(C2(F)CCC2)=O)CC1 c1(C(=O)NC2CCC(NC(c3ccc(-n4cncn4)cc3)=O)C2)cncc(F)c1 N1(C(C(=Cc2cnc[nH]2)C)=O)CC2CC(C1)C(CO)C2NC(C1CC1C)=O c1(C(N2C(C)CCC(NC(=O)CO)C2)=O)ccc2cc(Br)ccc2c1 C(CC(=O)NCC(C1CCCC1)NC(=O)CCSCCCC)=CC=C N1(C(C(C)(C)C2CCN(C(C3CCCN3C=O)=O)C2)=O)CCC12CCC(O)CC2 N1(C(c2c[nH]cc2C2CC2)=O)CC2CC1CN2C(C1CC2CCC2C1)=O N1(C(C(C)n2ccnc2)=O)CC(NC(c2ccc(C(F)F)cc2F)=O)C2CC2C1 C1(CNC(C(C)C#N)=O)CC(F)CN1C(=O)CC(c1ccccc1)N(C)C C(C(C)(C)C(=O)NCCCNC(=O)CC1CCCN1C(=O)OCC(C)(C)C)CC CCC(C(=O)OC)C(=O)N1CC(CCNC(=O)C(CC(C)C)NC(C)=O)(OC)C1 CC(C)C(CC(=O)NCC1=CCCN(C)C1)NC(c1ncc[nH]1)=O C12(c3cccc(C(=O)NCCc4cncc(C)n4)c3)CC(C)(C1)OC2(C)C c1(N2C(CNC(=O)C=Cc3cn[nH]c3)C(C3CC3)CC2)ncnc2cc(Br)sc12 c1(CC)cc(C(=O)NCc2ccoc2C(N2CC(c3cc(O)n[nH]3)C2)=O)ncn1 c1(C(C(=O)NC(C)CO)NC(COCCOC)=O)cccnc1 C1(C(=O)Nc2c(C)cccn2)CN(C)CCN1C(C1CCCO1)=O C1(CC)CN(C(c2cc(C)ccc2O)=O)CCN1C(=O)C1=C(Cl)CC1 c1(C(NC(=NCC)NCC(C)(C)COC)C)coc2c(F)cccc12 C(=O)(C(CC(F)F)N(C(=O)CC#N)C)N1CCC(CN(C)C)C1 C1(NC(CCC=CC)=O)CN(C(=O)C=C(C)C)CC(F)(F)C1 N1(C(C)=O)CCOC(C(N2CCC(NC(c3nnn(C)c3N)=O)CC2)=O)C1 C(=O)(C(C)(C)CC(F)F)NCC(CN(C(Cc1c(C)nn(C)c1Cl)=O)C)O c1(C(=O)NCCC2(CNC(C(CC)C)=O)CC2)ccc(OC)nc1Br N1(C(CC(C)O)=O)CC2CCCN(C(=O)CC3(C(F)(F)F)CC3)C2C1 c1(NC2CCC(c3nnnn3CCCF)(NC(=O)OCC)C2)cccc(Cl)c1Cl c1(N(C)CC2CCCN(C(C(c3c(C)n[nH]c3C)C)=O)C2)ncnc2sccc12 c1(C(N2CCCC(CN(C(c3cnc[nH]3)=O)CC)C2)=O)ncc2ccccn12 c1(C(N2CCCC(CNC(Cc3cc(C)no3)=O)C2)=O)nnn2c1C(=O)NCC2 [N-]=[N+]=NC1CC2(C(=O)NC3CC(NC(c4ncoc4-c4ccon4)=O)C3)CC12 c1(C(=O)NCCC(C)N(C(=O)C(O)Cc2ccccc2)C)ccc(C(C)(C)C)s1 c1(CC)nc(C)oc1C.C12(CCC1)N1CC(C(O)C(=O)NC2C)C1 CC(CCC(C)(C)C)C(=O)NCCC1CCCCN1C(=O)Cc1nncn1C CCCCC(C)C(=O)NCC1(OC)CN(C(C2(C)CCC23CCC3)=O)C1 C#CCCC(C(=O)N1CC(O)(CCC)C1)NC(C1CC=CCO1)=O C(=O)(C(C)(C)CC1CC1)NCCC(C)NC(=O)CC1CCC(=O)O1 C1(C(=O)NCCNC(C(CC=CC)CC)=O)CCc2nc(O)[nH]c2C1 CCCCC(O)CC(=O)N(C1CN(C(=O)Cc2ccnc(Cl)c2F)CC12CC2)C n1(CC)cnc2nc(=NCC3CC3(C)C)[nH]c(NCc3ccc(OC)c(C)c3)c12 C12CC3CC1CC3NC2=O.C1(CC(=O)OC)OCCCO1 N1(C(C(CC(CC)C)NC(c2cccc(F)c2)=O)=O)CCC2CN(C)CC2C1 C1(NC(C2(N(C)C)CC2)=O)CN(C(=O)CC2CCOCC2(C)C)CCC1CO CC1(C)CC(C(=O)NC2(C)CC2(C)C)N(C(C2CC3(CSC3)C2)=O)C1 C(C)(C(C(=O)NCCc1cscn1)NC(=O)CCc1nc(O)n[nH]1)OC C(=O)(C(O)CC[S+](C)C)NCCN(C(=O)C1=CCSC1)CCOC Cc1cc(C)c(NC(=O)CC2(N(C(=O)C=C(Cl)Cl)C)CC2)cc1O C(=O)(CCN=[N+]=[N-])NCC1(C(C)NC(=O)CCN2CCCCC2)CC1 c1(CC(=O)NC23CC(NC(C=C(COC)C)=O)(C2)C3)cn(C)nc1C c1(C(N2C(C)CC(CNC(c3cccc(CO)c3)=O)C2)=O)ccnc2[nH]cnc12 N1(C(C2(C=C)CC2)=O)CC2CCCC2(CNC(c2ccnnc2O)=O)C1 C(N=c1[nH]c(=NC(C)c2n[nH]cc2C(C)C)[nH]c2c1COC2)C1CC(OC)C1 N1(C(C(C)n2ccnn2)=O)CC2CCC1CN2C(C1CC1C1CC1)=O C1(OC)CCn2cc(C(=O)NC3CCCN(C(=O)CSC(F)F)C3C)nc2C1 c1(C(=O)NCC(CC=C)NC(c2cocn2)=O)nc2c(cc1Cl)OCCO2 C1(CCNC(COC2(C)CN(C(c3c(C)occ3)=O)C2)=O)CCCC1(C)C Cc1c(CC(=O)NC2CCC(CNC(C34CC(CO)(C3)C4)=O)C2)ncn1C C1(C(N(CC(CC)NC(C2(C)CC(C#N)C2)=O)C)=O)CCCC(=O)N1 CC(C)(Cc1cccc(Cl)c1)C(=O)NCCC1CC(NC(C2CC2CF)=O)C1 N1(C(C(C)n2cccc2)=O)CCCC(C)(CNC(=O)C=CCN2CCCCC2)C1 C(CN=C(NCC1CCC(c2ccccc2)O1)NC1CCC1)c1cc(C)no1 C1(NC(C2(COCC)CC2)=O)CC(C)CN(C(=O)CC2C=CS(=O)(=O)C2)C1 CC(C)(C)C(CNC(C1(C#N)CCC1)=O)NC(=O)C(=O)NCC1CC1 c1(C(c2c(C)onc2)NC(=O)Cc2onc(C)c2Br)cccc(O)c1 C1(C(=O)NCCCNC(c2cnn(-c3ccccc3)c2)=O)CCC(=O)N1C1CC1 C1(C(=O)NC(C(=O)N(C)CC)(C)CSc2ccc(C)cc2)CC2CC(=O)C1O2 Cc1ccc2c(NC(C3(C)CN(C(c4cc(F)c(C)c(F)c4)=O)C3)=O)n[nH]c2n1 N1(C(c2cc(C)[nH]c2C)=O)CCN(C(c2cnc(S)n2C)=O)C(C)C1C C1(CNC(CCCN(C)C(C2CC3CCC2CC3)=O)=O)CCCC2(CC2)C1 C=C(C)CCCC(=O)N(CCNC(=O)C(n1cc(Br)cn1)C)C1CC1 C1(NC(C2C(C)C2C)=O)CCN(C(c2ccc(Cl)cc2N)=O)C(C)C1 c1(C(=O)NCC(C2CCC2)NC(C2C(CC(C)(C)C)C2)=O)cn2ccnc2s1 C1(NC(Cc2c(C)n(C)nc2)=O)COC2(C1)CN(C(=O)C1=C(Cl)CCCC1)C2 Cc1sc(C(F)(F)F)nc1C(=O)Nc1cccc(NC(C2(C)COCCO2)=O)c1 N(C1CCCc2cc(CNC(c3ccon3)=O)ccc21)C(C1N(C=O)CCC1)=O C(=O)(C1c2ccccc2C(=O)N1C)N1CCC(CNC(C(CCOC)(C)C)=O)C1 c1(C(=O)NC2C(NC(C(C)O)=O)C2)cc(=NC(=O)OC(C)(C)C)[nH]n1C C1(C(=O)NCC(CN(C(=O)Cc2cnc[nH]2)C)O)CCC(C2CCC2)CC1 C(=O)(CS(F)(F)(F)(F)F)NC(C1OCCN(C(C(CC)(F)F)=O)C1)C c1(CC)nc(C(N2CC(C(C(=O)NC(C)Cc3ccccn3)OC)C2)=O)c(C)o1 CCCCCCCCNC(=O)CO.C1(OCC=CC)CCN(C(C2CCO2)=O)C1 O=C(C1=CCOCC1)N1CCC2C(C(N3CCOCC3C(F)F)=O)C2C1 N1(C(CNCC2CCC(c3n[nH]c(=N)s3)C2)=O)CCN(S(=O)(=O)CCCl)CC1 c1(C(c2ccoc2)NC(=O)NCCOC(C)=O)ccc(Br)cc1 c1(NC(C2CCC2(F)F)C)ccc(N2CCCC2=O)cc1 c1(C(N(C2CCN(C(=O)Cc3nc(=N)[nH][nH]3)C2)CC)=O)ccn(C(C)(C)C)c1 C1(NC(c2cccc3cnccc23)=O)CC2(CCCCN2Cc2ccccc2)C1 C1(C(N2CCC(CNC(C(CCSC)OC)=O)C2)=O)C2CCC3(COC(=O)C13)O2 C(=O)(CCCC(=O)N1CC(C(N)=O)(CNC(c2cn(CCOC)nn2)=O)C1)NC c1(C(N2CC(C(=O)Nc3cccc(C(=O)OC)n3)SCC2)=O)cc(F)cc(I)c1 N1(C(C(Br)=C(C)C)=O)CCCC1CNC(c1n[nH]cc1C)=O N1(C(C2CCC(C)(C)O2)=O)CCCC(C2CN(C(=O)CC(C)(O)C3CC3)C2)C1 N1(C(CC=C)=O)CCOC(C)(CNC(c2cccc(C(F)F)c2C)=O)C1 N1(C(C(C=C=C)C)=O)CC2(NC(c3ccc(S(N)(=O)=O)nc3)=O)CCCC2(F)C1 C(N=c1[nH]c(NC2CCCn3nccc32)nc2cccc(F)c12)C1(C)C(C)(C)C1 O=NN1CCCC1C(=O)NC1C2CN(C(c3ccnnc3)=O)CC12 N1(C(c2nc(COC)sc2)=O)CCC(C)C(CNC(=O)CCc2csc(=N)[nH]2)C1 C1(CN2CCC(NC(c3c(F)cc(C)c(F)c3)=O)C2)C2CC3CC(C2)CC1C3 Cn1nnc2c(NC3CC(CNC(=O)C(O)C4CC4)C3)ncnc12 C1(C(=O)Nc2c(C)cncn2)CC12CCN(C(=O)Cc1c(F)cccc1Cl)CC2 c1(C(N)=O)cc([N+](=O)[O-])cnc1NCC1CC2COCC2N1C(=O)COCC1CC1 C1(NC(c2c(CN(C)C)ccs2)=O)CCC(F)(CNC(C2CN(C(N)=O)C2)=O)C1 CCS(=O)(=O)CC(=O)N1CCC(C(=O)NCC(C2CCCC2)C)O1 Cc1cc(Br)c(OCC(=O)NC2CC2C(=O)NCCSc2ccccc2)c(Br)c1 C1(NC(CCCOC(C)C)=O)CCCCC1CNC(c1ccc(C(C)O)cc1)=O C1(C)(C(N2C(C)(C(C)C)CC2)=O)CCN(C(C2CC(O)C(F)C2)=O)C1 C1(NC(Cc2ccc(OC(C)C)cc2)=O)C(C)CCN(C(C2(SC)CC2)=O)C1C N1(C(c2csc(C3CC3)n2)C(=O)NCC2CC2)CCCC(F)(c2ccccc2)C1 c1(-c2cn(CCC)nc2)cc(C(=O)Nc2cncnc2OC)cc2cc[nH]c12 C1(NC(c2[nH]cc(C(=O)OC)c2)=O)CCCN(C(=O)CCC2CCC(=O)N2)C1C c1(OC)cc(C(=O)N(CCCNC(=O)CC2CCCC2)CO)ccc1S(N)(=O)=O N(C1CCCc2ccoc21)C(C1CCC(CNC(C(C(=O)OC)(C)C)=O)CC1)=O CC(CN(C)C)CC(=O)NCCCCNC(c1cnn(C)c1C1CC1)=O C(C(CC(F)(F)F)NC(c1cccc(C2CCOC2)c1)=O)NC(CNC(N)=O)=O CCC(C)(C(=O)NC1CCCC1NC(C1CC(F)(CO)C1)=O)OC C1(NC(C2(F)CN(C(C(C)N3CCCC3)=O)C2)=O)CCN2CCCC2C1 CC(C)C(C#N)C(=O)NC1CCCC(NC(c2cc(C#N)c[nH]2)=O)C1 CC1(C)NC(=O)N(CCC2CCCC2)C1=O.c12cc(ncn1)N1CCCC1CN2 C(CCCCCC=C)N(C(CCC#C)=O)CCNC(=O)CCS(C)=O c1(OCC)cc(C(=O)NCC2(C)CCCN2C(C2CN(C(C)C)C2)=O)oc(=O)c1 N1(C(c2c(OC)c[nH]n2)=O)CCCCC(NC(=O)Cc2csc(C)c2)C1 C1(C(C)NC(C=C(C)C(C)C)=O)CCCCN1C(=O)COc1ccccc1F C(CCC(=O)N1CC(N(CCO)C(c2ccc(Cn3cc(Cl)cn3)o2)=O)C1)=CC C(=O)(C(O)CC(C)(C)C)N1CCC(C)CC1CNC(=O)CC(=O)OC(C)(C)C Cn1c(C(N2CCCC(NC(=O)CCOCC3CC3)CC2)=O)cccc1=O CCC(CC)C(=O)NCC(=O)NC(CN(C)C(c1cnc(C)[nH]1)=O)CC c1(OC)cnc(C(=O)N(CCCCN(C)C(c2cnn(C)c2)=O)C)c(F)c1 C1(C(=O)NC2(CNC(C3(N(C)C)CC3)=O)CCOCC2)CCC2CC1CO2 C1(C(N2CCCCC2c2nc(C)cs2)C(=O)NCCCSCC)CC2CCC1O2 CCC(C(=O)NCC1CC(C)N(C(c2cc(N)cc(O)c2)=O)C1)C(F)(F)F C(CCN=C(NCC(C1CCCCC1)O)N1CCSC(C(C)C)C1)OC N1(C(c2cnc(CC)o2)=O)CC(NC(c2csc(S(N)(=O)=O)c2)=O)C2(CCC2)C1 c1(C(=O)NCc2cn(CC(N3CC(C#C)C3)=O)nn2)sc(C)cc1C C(CC(C(=O)N1CC(n2cnnc2)C1)NC(=O)CC(CC)C1CC1)OCC N1(C(Cc2cc(C)on2)=O)C2CCC(C(=O)NCC(=O)NC3CC3)C1CC2 N1(C(C(=O)NCc2ccc(-c3ccc(F)cc3F)o2)=O)CC2(CNCCO2)C1 c1(C(=O)NC2CCN(C)C2)cc2cc(F)c(F)cc2[nH]1.c12cccnc1C(=O)N2 C1(NC(C(CC2CCC2)NC(c2cscn2)=O)=O)CC2C(O)C(O)CC12 C1(C(N2C(C=C)CCC2)=O)CCCN(C(C2CC2(Cl)Cl)=O)C1C N1(C(c2ncn(CC)n2)=O)CC2(CCCC2)C1C(=O)NC1CCC(O)CC1 c1(C(=O)NC(Cn2cc(CNC(C(CC)C)=O)nn2)C)cc(OC)cc(F)c1 C1(C)(C(=O)NCC2N(C(C(C)Oc3ccccn3)=O)CC2)CCCC(F)(F)C1 c1(C(CC)C(=O)NC(CNC(=O)Cn2cc[n+](C)c2)C(C)C)ccc(F)cc1 Cc1c(C(=O)NCC(C)NC(c2nocc2Cl)=O)nn(C)c1N C12(NC(=O)C3=CCC3)CCCC1N(C(c1occ3c1CCCC3)=O)CCC2 c1(OCC(C)NC(=O)NCC(c2ccccc2)C)cccc2ccccc12 N1(C(C(C=C)(C)CC)=O)CC2(CCN(C(c3cncc(CC)c3)=O)C2)C1 c1(C(N)=O)nocc1C(=O)N(CCC(=O)N(CCC1CC1)CC1CC1)CCO Cc1ccc(C(=O)N(CCCN(C(=O)CN(C2CCSC2)C)C)C)cn1 c1(C(=O)NCC(CNC(C2OCCN(C(C)C)C2)=O)(C)O)c(N)ccc(F)c1F C1(C(N2CCC(Cc3cccc(OC)c3)C2)=O)CC2(C1)CC(F)C2 c1(C(=O)NC(c2cncs2)CF)cn2ccccc2n1 C(=O)(C(C(C)CC1CCCCC1)N1CCC(C(=O)NC)C(O)C1)NC N1(C(CSC)=O)CC2(NC(c3nccc4nn[nH]c34)=O)CCCC2(F)C1 C=C(C)c1cccc(NC(=O)CCOC2CN(C(=O)C=CC3CCOC3)C2)c1 O=C1CCC(C(=O)N2CCCC(O)(CNC(C3CC(C(F)F)C3)=O)C2)=NN1 N1(CC#N)CCN(C(=O)Cc2cnc(-c3ccccc3OCCO)cn2)CC1=O c1(C(=O)NC2CN(C(C(C(C)C)C)=O)CC2C(F)F)cc2c(Cl)c(Cl)ccc2[nH]1 N1(C(C2CCN(C)CC2)=O)CCC2CN(C(C3CCCN3C)=O)CC2C1 c1(CCC(=O)NCC2N(C(C3C(CC)C3)=O)CC(O)C2O)c(C)nc(O)nc1O O=c1c2cc(Cl)ccc2nc(O)n1Cc1nc(C2CC2)n[nH]1 C1(O)(C(N2CCC(C(C)(O)CNC(=O)CCC3CCC3)C2)=O)CCCCC1 c1(CC(=O)OC)onc(C)c1C(N1CCC(NC(=O)COc2ccccc2)C1)=O C1(NC(c2n(CC)nc(C)c2)=O)CC2CN(C(=O)C3=CCSC3)CCN2C1=O CC(C)C(C(C)NC(=O)CCc1ccccc1F)NC(c1ccnn1CCF)=O C1(C(N(C2CCCC2(F)F)C)=O)CCOCCN1C(C1CC(=C2CC2)C1)=O CCC(COC)C(=O)N1CCCC(CCNC(C23CC(C(C)C)(CO2)C3)=O)C1 Cc1n[nH]cc1CC(=O)N(C(C1CCOC1)CNC(=O)CC1(C)CCOC1)C1CC1 c1(C(c2n(CCO)nnn2)NCCCC2CCCCC2)ccc(F)c(C2CC2)c1 C1(C(=O)NC2(CNC(c3sccc3C3CC3)=O)CCOC2)CCc2ncsc2C1 Cc1ccc(NC(C2CC2C(=O)NCc2cccc(CO)c2)=O)c(F)c1 N1(C(CN2CC(C)C2)=O)CCCC(C2CCN(c3ncnn4cccc34)C2)C1 C(=O)(C(C)CC(F)(F)F)OC(=O)N(c1cc(C(C)C)nn1CCl)c1ccccc1 C(CCCCN=C(NCc1cn(C)nn1)N1CCCCC(C)(F)C1)SC C(=O)(CCCCC#N)NCC(C(=O)N(C(C)CC(F)(F)F)C)C C12(OC)CC(C(N3CCCC3(C)CNC(c3cc(C)nn3C)=O)=O)C(C1)C2 N1(C(C=CCN(C)CC)=O)CC(CNC(=O)C(C)(C)c2cccs2)C2(CCC2)C1 c1(N2C(C)C(NC(=O)CCn3cccn3)CC2)ccc([N+](=O)[O-])cc1Br C1(C(=O)NC(CN(C(=O)C=C2CCC2)C)(C)C)CCCC2(CCCCC2)C1 c1(C(=O)NCC2CC3(CN(C(C4(C)COCCO4)=O)C3)C2)cc2sc(Cl)cc2s1 C(CC(O)C(F)(F)F)NC(C(CN(C)C)NC(=O)COCC1CCCO1)=O N1(C(c2ccc(C(C)=O)[nH]2)=O)CCN(C(c2cc(C(C)(C)C)on2)=O)CC1CF c1(OCC)ncnc(OC)c1C(=O)NCC1CCCC1NC(=O)COC(C)(C)C c1(NC(C(=O)NCc2cc(Br)ccc2F)=O)c(F)cc(Br)cc1Cl Cc1ccc(C(c2nnnn2C2CCCCC2)Nc2cccc(Cl)c2C)c(Br)c1 C1(NC(C(C)NC(N)=O)=O)CN(C(=O)C(c2cnn(C(C)(C)C)c2)=O)CC1F c1(C(N2CC(C(=O)NC(C(CC)C)CO)C(F)C2)=O)ccc2nccn2c1 C1(C(=O)NC23CC(CNC(C(CC)NC(N)=O)=O)(C2)C3)CC12CCOCC2 N1(C(C(C)CS(C)=O)=O)CCOC2(CCN(C(c3cc4[nH]ccc4s3)=O)CC2)C1 c1(C(=O)NC2(CCCNC(C(COC)C)=O)CC2)cccc2c1CC(C)(C)C2 C(=O)(C1=CC2(CCOCC2)C1)NCCCCC1CN(C(C(CCC)N(C)C)=O)C1 CCC(C)C(O)C(C)C(=O)N1CCC(C)C(CNC(c2cnsc2C)=O)C1 c1(N(C(c2ccc(C(c3nc(C)[nH]n3)(C)C)o2)=O)C)ccc(C#N)cn1 C1(NC(C(N2CCOCC2)C)=O)(CNC(c2ccc(F)o2)=O)CCOCC1 C(=O)(C1(O)CCCc2ccccc21)C(C)(C)C.N12CC3CCC3(C1)OC2=O CC1COc2c(C(=O)N(C)CCOCCNC(C3(C)CC=CCC3)=O)cccc21 C1(C(=O)NCC(CC)NC(c2ccc(=O)oc2)=O)CCc2n[nH]cc2C1 c1(C(N(C)CC2(O)CN(C(C(COC)C)=O)C2)=O)nc(OC)ccc1F c1(C(=O)NCCC2(O)CCN(C(CCCCC)=O)C2)nn2c(c1Br)CCC2 N1(C(N2CCCC(C(N3CC4COCC4C3)=O)C2)=O)Cc2ccccc2C1 c1(C(=O)OC)ccc2nc1C(=O)N2.C(=O)(C(O)C(C)(C)C)N1C(CO)CCCC1 CS(=O)CCC(=O)N1CCC(C(C)(C)NC(=O)CSc2cccs2)C1 C12(NC(c3c(SC)csc3)=O)CCC(CNC(=O)CCC3CCCCO3)(C1)OC2 c1(-n2cc(C(CC(N)=O)NC(c3cc(Br)co3)=O)nn2)cc(Cl)cc(Cl)c1Cl C1(NC(CC(C)NC(C(n2ccc(C)n2)C)=O)=O)CCn2cncc2C1 N1(C(CCOC)=O)CCN(C(C)CNC(=O)C(COc2ccccc2)OC)CC1 C1(C2CCN(C(=O)C3=CCOC3)C2)(NC(c2cc(C(F)F)ccc2Cl)=O)CC1 N1(C(c2ccc(OCC)cc2)=O)CCC(C(=O)Nc2ccc(Cl)cc2O)C1(C)C C1(CC(=O)NC2CC(C)(NC(CCC(C)C)=O)C2)CC2CCC(C1)N2C c1(C(=O)NCC2(C(=O)NCC3(CC#C)CCCC3)CC2)c(Br)ncn1C N1(C(C2C(C)(C)NC(=O)C2)=O)CC(C2CCN(C(C3(C)CCCN3C)=O)CC2)C1 C1(CNC(C(C)(C)NS(C)(=O)=O)=O)CCCCCN1C(C12CC(O)C1C2)=O N1(C(C(CCC)F)=O)CCN(C(=O)CCC(C)CN(C)C)CC1C1CC1 N1(C(C(CC#C)C2CC2)=O)CCOCCC1C(N1CCC1CC)=O C=CC(C)(O)C(=O)NCC1(C(=O)NCCN2CC(CF)C2)CCCC1 C1(C(=O)NC2(C)CN2)CCCC1.C1(CCOCC)(C(=O)NC)CCC1 C1(C(=O)Nc2cccc(OCCC)c2)CC12CC(C)(C)C2 c1(C(N(C(C)C)CCNC(=O)C(C)S(N)(=O)=O)=O)ccc2cccc(F)c2n1 C1(NCCO)(OC(N)=O)CCOCC1.CC1CC(=O)N1.C12(CCCC1)CC(=O)N2 c1(CCNC(=O)C(=O)NCc2ccc(F)cc2)ncccc1CNC(CCC#C)=O c1(C(=O)NCCOCCCNC(c2n(C)nnc2)=O)coc2c1NC(=O)CCC2 c1(C(=O)NC2(C3CCCCN3C(C3CC3F)=O)CC2)cc(Cl)ccc1F C1(NC(c2c(C)nc(CO)s2)=O)CN(C(=O)Cc2cc[nH]c2)CC1S(C)(=O)=O c1(CN(C(C(=O)OC)CC(N)=O)C(c2ccccc2)=O)ccc2sccc2c1 c1(CNC(C2CCCC3CC23)=O)cnn2c1CN(c1ccn3nccc3n1)CC2 N1(CC2C(=O)NCCC2)CCCCC2(CCN(C(=O)C3=CCCCO3)C2)C1 Cc1cc(C(N2CCC(C)(NC(C3CCCN3N=O)=O)C2)=O)nc(N(C)C)n1 C1(C(N2CC(n3cc(CC(C)O)nn3)OCC2)=O)CC(C)(C)CC(C)(C)C1 C(CCCC(=O)NC(C)CC1CN(C(C2CCC2C)=O)C1)ONC(=O)OCCC=C C(=O)(C(F)C(F)(F)C(F)(F)F)NCC1C2CN(C(c3c(C)cccc3C)=O)C1C2 C#CCCN=C(NCc1c(O)cccc1F)N(C)CC1CC(OC)CN1C N1(C(CCc2cc(C)on2)=O)CCCC(F)(C(=O)N(C)CC2CCN(C)C2)C1 C1(C(=O)NCCn2nccn2)CCCC(NC(C2(CO)CCCCC2)=O)CC1 N#Cc1ncc(F)cc1NC(C1CC(O)CN1Cc1cc(F)c(I)c(F)c1)=O C1(C(=O)NCC2CN(C(c3c(CC)nccn3)=O)C2)CCC(=O)N(CCOC)C1 C1(CCO)(NC(=O)NC(c2ccccc2F)C(C)=O)CCC(F)(F)CC1 C(=O)(N=c1cc(C)o[nH]1)c1c(NC(CCc2nccc(C)c2)=O)cccn1 CCC(CCCC(=O)N1CCC(OC)C1C)NC(c1cnc(=N)[nH]c1)=O C(=O)(CCC(C)(C)C(=O)N(CC(C)NC(c1c[nH]nc1-c1cccs1)=O)C)OC Cc1cc(C)n(CC(N2CC(CCNC(C3(CCCF)CC3)=O)C2)=O)n1 N1(C(C(CC(C)C)C(N)=O)=O)CC(CNC(=O)CC(F)(F)F)CC12CCOCC2 c1(N(C2CCN(C(=O)CCCNC(=O)CC#N)C2)C)ccccc1 c1(C(=O)NCC2C3CN(C(C4CC5CC5C4)=O)CC23)cc2ncccc2[nH]1 N1(C(C)=O)CCC12CCN(C(c1sccc1C(N)=O)=O)CC2 CC(C)(F)CCC(=O)NCC1CCN1C(c1cnc(OCC2CC2)cn1)=O C1(CNC(C(C=C)(C)C)=O)CC2(CCN(C(=O)COCCOC)C2)CO1 c1(C(N(C)CC2CCCN(C(CCNC(=O)NC)=O)C2)=O)nccc(N)c1Cl Cc1c(C(=O)NC(C)(CNC(C2(CF)CC2(F)F)=O)CO)cnn1CCO C(=O)(CC1CNc2ccccc21)N1C(C#C)CNCC1 N1(C(C(c2ccc(F)cc2F)C)=O)CCCC(NC(C2(C)CCCS2)=O)CC1 C1(NC(=O)CCn2cccn2)CN(C(C2(Cl)CC2)=O)CC1n1cccn1 C1(CC(C)C)(CCCOCCN2CCOCC2)CCCN(C(=O)OC(C)(C)C)C1 c1(OC)cccc(CC(=O)NC2(CO)CN(C(=O)C(C)(C)C3CCCO3)C2)c1 c1(C(=O)NCC2N(C(CCS(C)=O)=O)CCC2)ccc(S(C)(=O)=O)o1 C1(N(c2nccc(C3CC3)n2)C)CCN(C(C2(n3ccnn3)CC2)=O)CC1 c1(C(=O)NCC(C)N(C(CN(C)Cc2ccc(C)cc2)=O)C)c[nH]cc(Cl)c1=O N1(C(C2C(CCC)C2)=O)CC(NC(c2cccc(F)c2OC)=O)CC(C)C1 C1(NC(Cc2c(C)ccnc2)=O)CC(C)CN(C(c2cc(C#N)oc2C)=O)C1 c1(COC)nc(CNC(c2nnnn2C(C)C)C2(CF)CCC2)cs1 C1(NC(C2CC(C)OC2)=O)(CNC(c2cc(N)nc(Cl)c2)=O)CCC(C)(C)CC1 Cc1cccc(C(=O)NCCC2C(C)CCCN2C(=O)CC(C)(C)C2CC2)c1C c1(C2(NC(=O)NCCC(C)NC(C(CC)C(C)C)=O)CC2)ccc2c(c1)OCO2 CCC(CNC(c1cc(O)ccc1F)=O)(CC)C(=O)N1CCC(CF)C1 CC1CC(CNC(C2CCC(F)CC2)=O)CN1C(c1ccsc1)=O C1(C(C)N(CCCC2CCC2)C)CCCC1 n1(CC)ncc(C(C(=O)NCC2CCOCC2)N(C)Cc2cnco2)n1 c1(CC)ccc(F)cc1C(=O)NC12CC1CN(C(=O)CCc1c(C)noc1Cl)C2 C(=O)(C(O)CC(F)F)N(C1C2CN(C(C3CN(C)C3)=O)CC21)C N1(C(c2n(COC)ncc2)=O)CCN(C(C2(C)CC(F)(F)C2)=O)CC(C)(F)C1 c1(C(=O)NC2CC(OCC(=O)N(C(C#C)C)CCCC)C2)ccn(C)c1 c1(NCCC2CC(=O)NC2)ccc2c(c1F)OCCO2 N1(C(=O)Cc2cc(C3CC3)on2)CCN(CCF)CC1 CN1CCN(CC(N2CCCC(N(C(=O)Cc3c[nH]nc3O)C)C2)=O)CC1 C(C)(CCCN=c1nc(N(C)CCN(C)C)c2[nH]ccc2[nH]1)SC C(=O)(C#CC(C)(C)CNC(c1cc(O)cc(F)c1)=O)NC1(C#C)CC1 c1(C(=O)NCC2N(C(CCN(CCCCOC)C)=O)CC2)cc(N)ccn1 c1(OC)ccc(S(=O)(=O)N2CC3(CCCC3)OCC2C(=O)O)cc1Br c1(C(=O)NCC(C)(C(C)C)NC(C(CC=CC)C)=O)ccn2ccsc12 C1(OC)CCN(C(c2ccc(-c3onc(CCOC(C)(C)C)n3)cc2)=O)CC1C N1(C(c2c(OC)cc(C)cn2)=O)CC(C)(C)CCC1CNC(=O)C=CC=C(Cl)Cl c1(C(=O)NCC(C)(C)OCCNC(C2CCCCC2)=O)occc1Br C1(C(=O)NC(CC=C)CNC(=O)CNC(=O)C(F)(F)F)C(F)(F)C12CCC2 n1(CC)ccc(C(N2CCC(OCCNC(C3CCC(O)CC3)=O)C2)=O)c1C C1(C(N2CCC3C(C(=O)NC(C4C5CC(=O)CC54)=O)C3C2)=O)CC2(CO)COC1C2 Cc1cc(CC(=O)NC2(CO)CCN(C(c3ocnc3C3CCC3)=O)C2)c(C)s1 c1(OC)cc(Cl)c(C)cc1C(=O)NC(CNC(c1cc2ccccc2s1)=O)CO O=C(C=CC=C(Cl)Cl)N=c1ccn(-c2ncccc2Cl)[nH]1 C1(C(=O)NC2CCC(N(C)C(C3CCCC34CC4)=O)CC2)(COC)CCC(=O)N1 CC1(CNC(=O)CC2CC(F)(F)C2)CCCN(C(C2CC=CCC2)=O)C1 c1(C(N2CC(CC(CNC(C(CC)(C)CC)=O)(C)C)C2)=O)nc2ccccn2c1F CC1CCOCC1C(=O)NCCCCN(CCCNC(C1CCSCC1)=O)C N1(C(CNC(=O)NC)=O)CC2(CCN(C(C3CC3c3cc(C)on3)=O)CC2)C1 N1(C(C(C)OC)=O)CCCOC(CNC(C23CC(C)(CO2)C3)=O)C1 C1(C(N(CCN(C(=O)CCS(C)=O)CC)CC)=O)CCC(C)(F)CC1 c1(COC(C(=O)NC(CN(C(c2c(OC)csc2)=O)C)C)C)cccc(C)c1 n1(CC(C)NC(C2(O)CCCN(Cc3ccccc3)C2)=O)nnc2ccccc12 C1(NC(COCC(=O)OC)=O)CN(C(C2CCC2)=O)CCC1C(F)(F)F C1(NC(C(C)(C)SC)=O)CC2(C1)CC(NC(=O)CCC(C)(C)c1ccccc1)C2 N1(C(c2c(F)ccc(N)c2)=O)CC(C2CN(C(=O)CCC3CCOC3)C2)C1 N1(C(CCN(CC)CC)=O)CC(NC(c2cnc(C(C)C)nc2C)=O)C2CC2C1 c1(CN2C(C(C)C)CN(C(=O)CC3CC4(CC4)C3)CC2)cc2ccncc2[nH]1 C(=O)(C1Cc2ccc(F)cc21)N1CCC(CNC(C=CC(=O)N(C)C)=O)C12CC2 C1(C(=O)NCC(=O)NCC#C)(CC)CCN(C(c2c(OC)cccc2Cl)=O)CC1 c1(CC(C)C(=O)N2CC(C)(NC(C34CC3COC4(C)C)=O)C2)ccc(Cl)c(Cl)c1 C#CCCCC(C)C(=O)NCc1cc[nH]c1C(=O)NC1CC1c1ccsc1 CC1(C)CCN(C(c2cc[nH]n2)=O)C1CNC(c1cnc(O)c(C(F)(F)F)c1)=O c1(C(C(=O)NCCN(C(C(COCC)C)=O)C)C)ccc2c(c1)OCCO2 c1(C(N2CCN(C(CCC=C=C)=O)CC2CCC)=O)cc2cc(C)ccc2[nH]1 C=C(C)CN=C(NCC(c1ccccc1SC)O)NC(C)CF C1(NC(c2c(CCC)n[nH]c2)=O)COC2CN(C(c3cnncc3OC)=O)CC12 N1(C(C)=O)CCC(N2CCN(CC(O)CC3CCCCC3)CC2)C2(CC2)C1 C1(C(N2CCC(=CCNC(c3ccccc3)=O)CC2)=O)CCC2(CC1)N=N2 c1(OC)cccc(C(N2CCC(O)C(F)C2)C(=O)Nc2ccc(F)cc2)c1F C12CCCCN(C1)C(=O)C(C(C)C)S2.c1(CC(OC)OC)cn(CC2CC2)nn1 c1(C(=O)NCC(C(C)C)NC(=O)C(C)(C)c2cc[nH]n2)ccc2ccncc2c1 C1(CCC)(NC(=O)CNC(=O)NC2CC2)CCCN(C(=O)C(Cl)=CCl)C1 C1(NC(c2csnc2Cl)=O)CN(C(c2cnn[nH]2)=O)C2CC12 c1(C(=O)NCCNC(c2cnn(C3CCOC3)n2)=O)cnn2c1CCCC2 C1(CCC)CN(C(c2c(Cl)cncc2Cl)=O)CCN1C(C1CC(=O)NC1(C)C)=O N1(C(CCCSC)=O)CCC2C(NC(c3cccc(OCC(C)C)c3)=O)CC12 c1(C(=O)NCC(C)(CO)NC(C(C)n2cncn2)=O)cc2n(n1)CC1(CC1)C2 N1(C(C(c2ccccc2)C)=O)CCC(N(C2CCN(CCO)C2=O)C)CC1.C(C(F)F)O c1(CCC(=O)NC2C(CNC(C(C)CN(C)C)=O)C2)ccc2c(c1)OC(F)(F)O2 N1(C(C=C(C)c2cccs2)=O)CCC(C)(C)C(NC(=O)C(C)Cc2cnc[nH]2)C1 N1(C(C(C)C)=O)C(C(=O)NC2CC(NC(N)=O)C2)C2CC(O)C1C2 c1(N2CCC(F)(CSC)CC2)nc(=NCc2cccc(Cl)c2F)[nH]c2c1COC2 N1(c2n(CCOC)c(-c3ccc(C)o3)nn2)CCC2(CC1)C(=O)N2.C(C)(C)OC c1(OC)ccccc1CC(=O)N(C)CC1CN(C(C2(O)CCOCC2)=O)C1 CC(C)CCC(F)C(=O)NCCC1CC(F)(F)CN1C(=O)C=CCO CC1(NC(=O)C(F)CC2CCOC2)CCN(C(=O)C2=CCCC2)C1 CC1CC(NC(=O)C=Cc2cccc(Br)c2)CCN1C(=O)C(=O)NCC1CC1 C1(C(N2CC(C)C(NC(c3ccc(Br)s3)=O)C2)=O)CC2(CCOCC2)CO1 c1(OCC(=O)NCC2CCCN(c3snc(CC)n3)C2)ccc(C(C)=O)c(C)c1 C1(NC(CCC(=O)OC(C)(C)C)=O)CC(O)CN(C(c2ccccn2)=O)C1 N1(C(CC2CCN(C(C3N(C(C)(C)C)CC3)=O)CC2)=O)CC(=O)NCC1C(N)=O C(CCCC(CO)NC(=O)CN1CCCC(CC)C1)NC(C(CCC)O)=O CC1(CN)CCCN(C(=O)C(N2CCN(c3ccc(O)cc3)CC2)=O)C1 CC1=C(C(=O)NC2CCN(C(c3c[nH]nc3F)=O)C(C)C2)CCCO1 CC(C(=O)NCCCN(C(C1(Br)CC1)=O)C1CC1)n1ccnn1 N#CC1CN(Cc2cc(F)cc(Cl)c2)CCN1C(c1ccc(CBr)cc1)=O N1(C(C(N)=O)=O)CC2CS(=O)(=O)CC2(NC(C2CC=CCO2)=O)C1 c1(NC(c2c(F)ccc(C)c2O)=O)sc2c(c1C(N1CCOCC1)=O)CCCC2 C1(NC(CC(CC)C2CCC2)=O)CC(OC)CN(C(=O)C(C)(F)F)C1 c1(C(NNC(C2NCC(CC)OC2)=O)=O)cc(Br)cc(N)c1C N1(C(C(C2CN(C(C3CC3(Cl)Cl)=O)C2)OC)=O)CCOCC(C)(O)C1 Cc1c(C(=O)NCC(CC(C)C)NC(=O)C=Cc2ccccc2)cc(O)cc1N N1(CC)CCN(C(C2(c3ccccc3)CCN(C(=O)OC(C)(C)C)C2)=O)C(C)C1 c1(OC)cc(Cl)c(C(=O)NC2CC(NC(c3cncc(Br)c3C)=O)C2)cc1OC N1(C(Cc2ccc(OC)cc2)=O)CCC2CN(C(=O)Cc3coc(C)n3)CC12 c1(C(N2CCCC(CNC(C=C(CC)CC)=O)CC2)=O)n[nH]c2c1CC(C)CC2 C1(OC)CN(C(=O)CCc2ccc(C)cc2)CC1NC(c1coc(C(C)=O)c1)=O N1(C(CC(CCC)O)=O)CC2(C1)CN(C(c1cnn3c1CC(C)CC3)=O)CCO2 c1(C(N2CC(COC)(NC(C(=O)NCCCOC)=O)C2)=O)cccc([N+](=O)[O-])c1 CCCCC(F)C(=O)N1CCCCCC1CNC(C12COCC1C2)=O c1(C(=O)NCC(C(C)C)(C)NC(C2CN(S(C)(=O)=O)C2)=O)cc(N)c(Cl)c(O)n1 N1(C(COCCOC)=O)CCN(C(c2noc(C)n2)C)CC1C CCC(CC(=O)N1CC(CN(C(=O)CCc2cc(C)no2)C)C1)C1CCC1 C1(N(C(C(c2cccs2)SC)=O)C)CN(C(=O)Cn2cc(C)cn2)CC12CC2 C1(NC(NC(c2sccc2C)CC)=S)CC(C(F)(F)F)CC(C(F)(F)F)C1 c1(CN(c2cc(NCc3ccccc3C#N)nc(C)n2)C)ccnc2[nH]ncc12 C(c1cc2ccccc2o1)=CC(N1CC(N(C(CC2ON=C(C)C2)=O)C)C1)=O CCCCC(CN=c1[nH]c(C2CC2)nc(=N)[nH]1)NC(=O)C=CC(C)(C)C C1(C(=O)Nc2n(C)nc(C3CC3)c2)CC2CCC1N2C(C1CC1(F)Cl)=O c1(C(=O)NCC2N(c3nc(OC)nc(C)c3)CCC2C)ccc2nccnc2c1 Cc1ncc(N)cc1C(=O)N(C1CCCC1)CCCNC(=O)C(C)C(C)O C1(NC(c2n3c(nn2)SC(=C)C3)=O)CN(C(c2cocc2C)=O)C2CCCCC12 N1(C(c2nc(NC(C)=O)sc2)=O)CCC2(CCN(C(=O)CC3=NNC(=O)C3)C2)C1 C1(C(=O)NCCCC(=O)OC)CCN(C(C2OCCC2C)=O)C1(C)C C(C(CNc1ccccc1)S(C)(=O)=O)NC(NC(C=C(C)C)(C)C)=O N1(CC(=O)NCC(CNC(Cc2ccc(OCC)cc2)=O)C)CC(=O)N(C)C1=O Cc1nn(CC(=O)NCC2(C)CCN(C(C3COC(=O)O3)=O)C2)cc1Br N1(C(C(C)(C)C(N)=O)=O)CC2(C(N3CC(c4nn[nH]n4)C3)=O)CCC1CC2 C1(NC(C2C(C)C2(F)F)=O)CCC12CN(C(c1ccc(F)s1)=O)C2 CCCCCC(O)CC(=O)NCC1COC(C)(C)CN1C(C1CC(N(C)C)C1)=O CC(C)(C)C(=O)CCC(=O)NC(CO)C(=O)NCC(c1ccncc1)O c1(C(N2CCCC(N(C(C(CC#C)C)=O)CCF)C2)=O)cc(C)ccc1NCC Cc1cn2c(C(=O)NC(C)CCN(C(=O)C=Cc3cc[nH]c3)C)c(Cl)nc2s1 c1(C(N(CC(C)NC(C2(SC)CC2)=O)CC)=O)ccc(O)nc1C N1(C(CC(COC)C)=O)CCC(C)(C)C1CC(=O)NCCOc1ccncc1 c1(OC)cncc(CNC(=O)CC2CCCN2C(=O)CC2CC(SC)C2)c1 N1(C(C2C(C)(C)C2)=O)CCOC(C)(CNC(C2CCC(CO)CC2)=O)C1 C1(CCNC(=O)CC2CCCO2)CCCN1C(c1cncs1)=O c1(C(N2C(C3(NC(C(C(C)C)F)=O)CC3)CCC2)=O)ccc2nn[nH]c2c1 N1(C(c2c(CC)cns2)=O)CC(OC)C(C(=O)NC2CCC(NC(N)=O)C2)C1 N1(C(C=CC(C)(C)SC)=O)CCC2CC2(C(N(C)CP(C)(C)=O)=O)CC1 C1(NC(C(C)CF)=O)CN(C(C2CCN(CC3CC3)CC2)=O)C2(CCCCC2)C1 C(CC(O)C(=O)N1CCC1(C)C)NC(C(C)c1ccco1)=O C1(OC)CCCCC1C(=O)NOCCCCC(=O)N1CCC1C1CCCCC1 CON(CCC(=O)NC1CC(CS(C)(=O)=O)C1)C(=O)CC1=CCCCC1 C1(C(=O)NCC2CCN(C(c3ncn(C)c(=O)c3)=O)CC2)CCC2(CCOC2)O1 N1(C(c2cccc(CC)c2C)=O)CC2CCC(C1)N(c1nc(C)ncc1F)C2 C1(CC(N2CCCN(C(C3CCOC3)=O)CC2)=O)CCc2ncc(Br)n2C1 CC1CC2CN(C(=O)CCC3CCC3)CC2N1C(c1ccc(Br)s1)=O N1(C(C2N(C(c3c(C)n(C)nn3)=O)CC=CC2)=O)CCN2CCC1C2 C(=O)(C1=CCc2ccccc21)NC1CCC(NC(c2c(CC)c(C)sc2)=O)C1 N1(C(CC2C(C)CC2)=O)CCCC12CCN(C(c1ncc3n1CCCC3)=O)CC2 c1(C(N2CCC(CCC(=O)NCC(C(C)(C)F)(C)F)C2)=O)c[nH]c2nccc-2c1 C1(C(=O)NCCNC(C2C3CCC2(c2cccnc2)C3)=O)C(F)(F)C12CCC2 N1(C(COCC)=O)CCC(C)C(CNC(=O)Cc2ccncc2Cl)C1 CCC(C)(C(=O)N(CC(C)CNC(c1cc(C)n(C)n1)=O)C)C(N)=O N(C(=NCCC(C)C)NCC1COC(=O)N1)C1CCN(C(CC)=O)C1 c1(C(C)C)ccc(C(=O)NC2CC23CC(NC(=O)CC2CCCNC2=O)C3)cc1 N1(C(C(C)NS(CC)(=O)=O)=O)CCN(C(=O)CCc2cccnc2C)C(CO)C1 c1(C(N2CC=C(CNC(C3CC(C(C)(C)C)C3)=O)CC2)=O)ccc(C#N)c(F)c1 C(CC(C)C(=O)N1CCC(NC(=O)CN(C)C(=O)C2CC2)CC1)OC C(C#CC(=O)NCC1CN(C(=O)C2CC2)C1)NC(C(C)NC(N)=O)=O C(=O)(C1=CC2CCCC12)N1CCC(NC(c2cc(F)ccc2F)=O)(CF)C1 C(=O)(CCCCC(C)=O)N1C(C(=O)NCCC(CCC)O)CSCC1 N1(C(C(C)Oc2ccccc2)=O)C2CCC1CN(C(C1CCN1S(C)(=O)=O)=O)C2 c1(C(N2CC(C(C)NC(CC3(CC=C)CCCC3)=O)C2)=O)ccc(OC)c(Cl)n1 N1(C(CCCC(=C)C)=O)CCC2(CC1)CN(C(=O)CCC1(C)CC1(F)F)CCO2 C(=O)(CCC(C)(C)F)N1CC(C(N)=O)(CNC(CSc2ccc(C)cc2)=O)C1 C1(NC(C2C(C)CCOC2)=O)CC2CCC1CN2C(C1(C)CCC1)=O Cc1cc(C)n(-c2cc(-c3nc(C4CC4F)n(CCCCO)n3)ccn2)n1 C1(NC(=O)NC2(C)C(C)(CNC(=O)OC(C)(C)C)CC2)CCS(=O)(=O)C1(C)C N1(C(c2c(CC)ccs2)=O)CCC(CNC(c2ncoc2C)=O)(COC)C1 C12(CNC3CCCN(C(C)C)C3)C(N)C3CC1C2C3 c1(CNC(COCCOC)=O)ccccc1CN(C)C(c1cncn1C)=O Cc1cn(C)cc1C(=O)NCc1cccc(C(=O)NOC2CCOC2)n1 C1(NC(c2ncoc2C(F)(F)F)=O)CN(C(=O)C2=C(Cl)CC2)C2CCCCC12 N1(C(C2CCCN(C(N)=O)C2)=O)CCN(C(=O)CCSC2CCCC2)C2CCC12 C1(CNC(Cc2c(CC)con2)=O)CC(OC)CN1C(=O)Cc1csnc1C N1(C(c2c(C)nn[nH]2)=O)CCCC(C2CC2NC(C2(C)CCCNS2(=O)=O)=O)C1 N1(C(C(=O)Nc2ccc(C(C)(C)C)c(Cl)n2)=O)CC2CC3CCCN3C2C1 C(=O)(N1CC2COCC2O1)C1N(C(CCC(CC)=O)=O)CC=CC1 c1(C(N2CCC(=CC(=O)NCc3nn[nH]n3)CC2)=O)cc(Cl)c(Cl)c(Cl)c1 C12(CCN(C(=O)NCC3Cc4ccccc4O3)C3CC3)CC3CC(CC(C3)C1)C2 CC1(C)Cc2[nH]nc(C(=O)NC3(C)CC(NC(=O)Cn4ncnn4)C3)c2C1 Cc1ccc(OCC(=O)NCC(C)(CO)NC(c2cc(CCO)on2)=O)c(F)c1 N1(C(c2cccc(OC)c2)=O)CCCC(NC(=O)C(N2CCC(O)CC2)C)C1C C1(NC(CN(C)C)=O)C(NC(CC2(NC(c3ccsc3)=O)CC2)=O)C1(C)C Cc1cc(CC(N2CC(NC(C3COCCO3)=O)C2)=O)no1 c1(OC)cc(C(=O)NCC2COC(CNC(C3CCCCC3O)=O)C2)cc(C)n1 c1(CC(=O)N(C2CCCCC2)CC(=O)OCCNC(C)=O)cncn1CO.CO C1(C(=O)NCC2CC(NC(c3nc(CC)[nH]n3)=O)C2)CCC(C)(C)CC1 C1(NC(c2c(CC)non2)=O)CN(C(=O)CSC(F)F)CC1C c1(C(=O)NC2CC(C)(C)N(C(=O)COC3CC3(F)F)C2)cc2cccn2cn1 c1(N(C)C)ccc(CNC2CC(C(=O)NCc3ccc(F)cc3Br)C2)c(O)c1 C1(CC)C(NC(=O)CC2CCCSC2)CCCN1C(=O)CCN(C=O)CCO Cc1cc(C(=O)NCc2cc(C(N3CC(C(C)(C)O)C3)=O)co2)nc(O)c1 C1(C(=O)NCC(C)NC(=O)OC(C)(C)C)CCN(C(c2c[nH]c(Br)c2)=O)C1 C1(SC)CN(C(=O)Cc2cccnc2)CC1NC(C1CC1c1ccncc1)=O N1(C(CC2(OC)CCCC2)=O)CCC(NC(=O)C(F)=C2CCC2)C(C(C)C)C1 Cc1ccc(C#N)cc1NC(C)(CCc1ccccc1F)c1nnnn1C1CC1 c1(C(=O)OC)c(C(=O)NCCC(C)(C)CNC(=O)C(CO)N(C)C)cnn1C c1(C(=O)NC(C2C(C(=O)NCCSCC)C2)=O)cc2cc(F)ccc2s1 n1(-c2ccc(C)cc2)[nH]nnc1=NC(C)C1CCN(C(c2coc(C)c2)=O)C1 N1(C(C(=CC2CCCC2)C)=O)CC(C2CCN(C(C3CCCN(C)C3)=O)CC2)C1 N1(C(C(C(C)C)OCC)=O)CCCC(CNC(c2n[nH]c3c2CCC3)=O)CC1 C1(CC)CCC(C(=O)NCC(N2CCN(C(=O)C(F)=CC3CC3)CC2)=O)CC1 C=C=CC(C)C(=O)N(C(c1ccccc1)CNC(c1cnn(C(F)F)c1)=O)C C12(NC(c3sc(C)c(O)n3)=O)CCC(C1)N(C(C1(CO)CCCO1)=O)C2 C12(CNC(c3cn(C)nn3)=O)CCCC1CCN2C(c1cc2c([nH]1)CCOC2)=O c1(COCC(=O)NCC(CNC(=O)COC2CCOC2)O)ccc(Br)cc1 Cc1cc(Cl)c(C(=O)NCC2CCC(NC(c3cc(C4CC4)on3)=O)C2)cc1F C1(NC(c2c(C(C)C)n(CCO)nc2)=O)CN(C(c2coc(O)n2)=O)CCC1CO n1(COC)nc(C(=O)N(C)CCN(C)C(c2cc(Cl)cs2)=O)ccc1=O c1(C(N2CC3C(C(=O)NCc4cnccn4)C3C2)=O)cccc([N+](=O)[O-])c1I c1(C(C)C)cc(NC(N2CCC(c3ccc(Cl)nc3)CC2)=O)cc(C(F)(F)F)c1 CC1CC(NC(c2cnoc2-c2cccs2)=O)CN1C(=O)COC1(C)CCC1 C12(CNC3CC(NC(C4(c5ccc(F)cc5Cl)CC4)=O)C3)CC=CCN1CCC2 c1(CCC)cc(C(=O)NCc2ncnn2CCF)ccn1 N1(C(C2C(=C)CC2)=O)CC=C(CCNC(=O)CCC(=O)N2CCOCC2)CC1 C=C(C)CC(C(=O)NC(CC)CC(=O)OC)NC(c1ccn(C)n1)=O c1(C(N2CC(O)(CNC(Cc3n(C)cnn3)=O)C2)=O)c(F)ccc2nc[nH]c12 C1(NC(C=CSC)=O)C2CCN(C(C3(c4cccs4)CC3)=O)CCC12 N1(C(CCc2cnc(C)s2)=O)CCOC(CNC(=O)C(c2cn(C)nc2C)C)C1 CCCC(C(O)C(=O)NCC1(C)CCN(C)C1)NC(C1CCC1OCC)=O c1(NC2C(C)CN(C(=O)CN3CCCCC3=O)C2)nc2c(cc1C#N)CCCC2 CC1(C)C(C(=O)OCc2nc(Cc3ccccc3)no2)CC12CC(=O)C2 c1(C(N(CCN(C)Cc2nc(C)[nH]n2)C(C)C)=O)c2ccccc2nn1C N1(C(c2cccc(C3CCC3)c2)C(=O)NC)CCC12CCC(C)(C)CC2 C#CCC(C(=O)N(C1CCOCC1C)C)NC(=O)CC(C)O Cc1c(Cl)ccc(C(N2CCC(=CC(=O)Nc3cc(F)c(Cl)cn3)CC2)=O)c1Cl c1(NC(C(=O)NCCCCC#N)=O)ccc2c(c1)CCCC2O c1(-c2c(CC)cco2)nc(-c2cccc(F)c2)nn1CC(=O)O N1(C(c2n(CC)nnc2)=O)CCN(C(C2(C(N)=O)CCC2)=O)CC2CCCCC12 c1(CC)ncncc1C(N1CC(NC(=O)CCC(C)N(C)C)C(CO)C1)=O CC1COCCC1C(=O)NCCC1(NC(=O)COCCc2ccsc2)CCC1 N1(C2CN(C(C3CC(Cl)(Cl)C3)=O)C2)CCN(C(C2(O)CCOC2)=O)CC1 N1(C(c2ccns2)=O)CC(NC(C23CCC(C2)C3)=O)C(O)C1 c1(C(=O)NCC(CNC(c2cc(C(=O)OC)no2)=O)OC)cncc(C(C)C)c1 c1(C(N2CC(NC(c3ccc(OC)cc3)=O)C(C)C2)=O)cc2ccoc2cc1F N1(C(C(=O)N(C)C)=O)CCC2(CC1)CCN(C(C13CCOC1CCOC3)=O)C2 c1(SC)ncc(N)c(C(=O)N(CC(C)CNC(C2CNC(=O)N2)=O)C)n1 CCCCC(CNC(=O)Cc1cccc(F)c1)NC(c1ocnc1C1CC1)=O c1(C(=O)NCC=CCNC(c2cncc(OC)n2)=O)ccc(S(=O)C(C)C)cc1 C1(NC(c2cc(C)ncc2)=O)CC12CCN(C(c1cc(N(C)C)cc(F)c1)=O)C2 C1(CC(N2CC(CCNC(c3cnc(N(C)C)o3)=O)C2)=O)CC2(CCC2)C1 C=C1CCN(C(=O)CC2CCCCCC2)C(C(=O)Nc2ccc(F)nc2OC)C1 C1(C2CCCN(C(c3cc[nH]n3)=O)C2)(NC(c2cc(OC)ncc2Cl)=O)CC1 c1(CC)conc1C(=O)NC1CC(CNC(c2cnc(C(C)C)[nH]2)=O)C1 c1(C(=O)NCC(C)CNC(C2(Br)CC23CCC3)=O)noc2c1COCC2 c1(C(N2CC3C(CNC(c4n(C)cnc4)=O)(C3)C2)=O)cc(=O)cc(Cl)[nH]1 N1(C(CCn2c(C)nc(C)n2)=O)C2CCC1(CNC(=O)CC1CCCC1O)CC2 c1(C(=O)NCC(C)NC(=O)Cc2cnco2)ccc(S(C)(=O)=O)[nH]1 Cc1ccccc1S(=O)(=O)CC(=O)N1CC(C2CCCN(C(C3CC3C)=O)C2)C1 c1(C(=O)NCC(C)N(C)C(c2ncccc2F)=O)cc(Cl)cc(Br)c1N C(=O)(C(F)(CNC(C1CCC1C)=O)C(C)C)NCc1cc(OC)ncn1 CCC(CNC(=O)CN1CCOC1=O)(CC)C(=O)NCC(C)(C)CO c1(C(=O)O)cn2c(n1)CN(C(=O)CC1(Cc3ccc(Br)c(Cl)c3)CCC1)CC2 N1(C(C(C)CF)=O)CC(NC(=O)C=Cc2cncs2)CC12CCC2 C1(CC#C)(C(=O)NCC2CCC(CNC(=O)CC3C=CCC3)CC2)CCOCC1 N1(C(C(=O)Nc2cccc(OC(C)C)c2)=O)CCS(=O)(=O)C(CO)C1 CC(C)C(C(=O)N1Cc2ccccc2CO1)NC(C1CCCC(C#N)C1)=O S(=O)(=O)(c1ncccc1C(F)F)NC(c1ccc(C)cc1C)C C=CC(CCC)CC(=O)NCCCCCNC(=O)C(C)(C)c1cccs1 C(=O)(C(C)(C)C(C)(C)O)NCC1(F)CC(CNC(c2cnc(C)nc2)=O)C1 c1(OC)cc(C)cc(CNc2c[nH]nc2C(=O)N=c2cco[nH]2)c1O c1(C(=O)NCC(C)N(C(CC2CC(=C)C2)=O)C)ccc(F)c(C)c1C c1(CC)c(C(=O)NCCNC(C2CC2C(=O)NC(=O)OC)=O)cnn1C C1(CNC(C2CCC3(CC3)N2C(=O)CCc2cn[nH]c2)=O)CC2CCCC2C1 C1(C(N(C2CC2)CC2N(C(CCC(=C)Cl)=O)CCC2)=O)CC(F)(F)C1(F)F CC1(c2cn(CC3(CC(=O)O)CC3)nn2)CCN(C(=O)CN2CCSCC2)CC1 c1(C(N(CCOC)CCOCCC(=O)NCC(C)(C)C)=O)cc(C)c(=O)n(C)c1 c1(C(C)C)ncc(C(=O)NCc2cn(C3CN(C(C4CC4F)=O)C3)nn2)[nH]1 C(C(=O)NCC1(n2nccn2)CC1)(C1CCCO1)NC(c1ccoc1)=O CC(C)C(CC(=O)N(C)CCOCCO)NC(=O)Cc1ccc(O)nc1 C1(NC(c2cc(C3CC3)ns2)=O)C2CN(C(C3CCCS3)=O)CC12 C1(CNC(CNS(CCCC)(=O)=O)=O)CCC2(CN(C(=O)C(F)(F)C3CC3)C2)O1 C(=O)(CC(C)(C)C)NC1CC(CCNC(C(C)Cc2cnn(C)c2)=O)C1 C1(CCC(=O)NCC2CC(=C)C2)CCN(C(=O)CCc2nncn2C)C1 c1(C2CN(C(=O)CSC3CC3)C2)cn(Cc2cccs2)nn1.c1(CC(=O)N)ccc(Cl)[nH]1 N1(C(Cn2c(=O)sc(C)c2C)=O)CCC2CCN(C(c3ccnnc3)=O)CC2C1 C(=O)(C(CC(C)(C)C)OC)N1C(CC)C(C(N2CC(C(C)(C)C)C2)=O)CC1 C(=O)(C(CC(C)C)N(C)C)NC1CC(NC(C2(OC)CC2)=O)CC1O O=C(C1=C(Cl)CCC1)NC1CC(F)CN(C(=O)C(F)CC2CCOC2)C1 C1(CNC(c2cnc(C)[nH]2)=O)N(C(c2cnc(F)c(Cl)c2)=O)CCCC1(C)C c1(C(=O)NC2C(CNC(CSC)=O)CC2)ccn(CC(F)F)c(=O)c1 Cc1cc(C)c(CC(=O)NC2CCN(C(=O)C(F)C3CCOC3)C(C)C2)c(O)n1 C(=O)(C(C(C)C)NC(c1cnns1)=O)NC(CCN(CC)CC)C Cc1cc(O)ncc1C(N1CCC(C(=O)OCCNC(=O)C(F)(F)F)C1C(C)(C)C)=O N1(C(C2CC(SC)C2)=O)CC2CC(C)N(C(=O)CC3CC=CCN3C)C2C1 CC1(C)CN(C(=O)C(=O)C(F)(F)F)CCC1NC(c1cc(-c2ccco2)no1)=O c1(C(N2CC(NC(C(C)CC#N)=O)(CF)C2)=O)cc2n(n1)CCCO2 C1(C(=O)NC(C(=O)NCc2c(C)nco2)CCC2CCC2)CC(C(C)C)=NO1 Cc1ccnc(C)c1C(N1CC(NC(C23CSC(C2)C3)=O)CC(O)C1)=O CN1CCC23CCN2N2CCC(C3C2(C)C)C1=O C(CC(C(=O)NCC1CN2CCC1C2)NC(c1cnnc(O)c1)=O)OC C1(CN(C(=O)Cc2ccc(Cl)cc2)C)COCCN1C(=O)C(O)C1CC1 CC(C(C)(C)O)N(C(=O)C(O)C1CN(C(=O)Cc2cncn2C)C1)C C1(NC(CCSCCC)=O)CN(C(c2cc(C)c[nH]2)=O)CC2(CCOCC2)C1 N1(C(C=C(CC)C)=O)CCCN(C(c2cnc(S)nc2)=O)CC1CO c1(OC)nc(NC(N2CCC(F)(c3cnn[nH]3)C2)=O)sc1C N1(CC)CC(N=c2[nH]c(N3C4C=CCC3CC4)nc3c2CCCCCC3)CC1=O N1(C(c2c(SC)nccn2)=O)CCN(C(=O)CC(C)(C)c2ccccc2)C(C)C1 C1(N(CCCc2cscn2)C)CCN(C(=O)CC2CCOCC2)C1 c1(CC)cc(F)c(C(=O)NC2CC(NC(C3CCCC(C)(C)O3)=O)C2)cc1F C(c1ccccc1F)=CC(=O)N(C)CC1CCN(C(c2n(C(C)C)nnc2)=O)C1 C12(C(=O)NCCOC3CCN(C(C(C)(C)OC)=O)C3)CCC(CC1)C2(C)C C1(C)(CNC(C2(CC=C)CC2)=O)CN(C(=O)Cc2cc(Cl)cc(Cl)c2)C(C)(C)C1 c1(CCC)c(C(=O)NCC2CCCC(CNC(c3cc(O)cs3)=O)C2)nnn1C C1(C(N(c2cccnn2)C(C2(c3nccs3)CC2)=O)=O)CCCN(CCCO)C1 C#CCC(CC(=O)NC1CC(O)CC1O)NC(=O)C=CCN(C)CC N1(C(CSC(C)(C)C)=O)CC2CCN(C(C3CC(CC4CC4)C3)=O)CC12 C(=O)(C(C(C)(C)C)NC(c1cnsn1)=O)NCC1(CCC)CCC1 C12(C(=O)NCc3ccc(CC(C)NC(=O)C(C)(C)C#N)cc3)CC(C1)S(=O)(=O)C2 N1(Cc2c(C)cccc2Br)CC2CCN(C(C3CCCCN3C)=O)CC2C1 N#Cc1ccc(NC(C2CC23CCN(S(=O)(=O)c2ccc(Br)s2)C3)=O)c(F)c1 Cc1nc(-c2cn(CC3CCCC3NC(=O)CCC3CCCCO3)nn2)sc1C c1(CCN(c2nnnn2CCN2CCOCC2)C(C2CCCS2)=O)cn(C2CC2)nn1 c1(N2CCN(Cc3cc(C(=O)OC)n(C)n3)C(C)C2)ncnc2occc12 c1(C(=O)NCC2C(NC(CCOC)=O)CCC2)c(C)coc1C1CC1 Cc1ccn(C)c1C(=O)NCc1nocc1C(=O)NCc1cnn(CCF)c1 c1(CC(=O)NCc2cn(C3CN(C(COC)=O)C3)nn2)ncc(F)cc1F CC(CC(F)F)C(=O)N1CC=C(C(=O)NC2CC3(CCCC3)C2)C1 c1(C(N2CCC(C)(NC(C3CCCC(C(C)(C)C)C3)=O)C2)=O)n[nH]c2c1COC2 c1(C(C)C(=O)NC2CC(C)(NC(C3CCOCC3)=O)C2)cc(Br)ccc1F N1(C(C2CC(=C)C2)=O)CCC(CNC(c2ccncc2C(=O)OC)=O)C12CC2 c1(NCC2N(C(CCCC#C)=O)CCC2)c([N+](=O)[O-])c(=O)n(C)c2ccccc12 Cc1ccc(C(=O)OCC2COC(CNC(=O)NC(C)(C)C)C2)c(C)c1 Cc1oc(C(=O)NCC(C2CCC2)NC(c2cnccc2Cl)=O)cc1S(C)(=O)=O C1(C)(C(N2CC(C)(NC(Cc3nc(COC)sc3)=O)C2)=O)CCOC1C C(=O)(C(C#N)(CC)CC)NC(CCC(N1CC(C=C)OCC1)=O)CC c1(NC(N2CCC(C(F)F)C2)=O)ccc2c(c1)OCCCO2 C(=O)(C(CO)C(F)(F)F)N1CCC(CC)(NC(=O)Cc2cscn2)CC1 N1(C(C(CC)SC)=O)C(C(=O)NC2CCOCC2OC)CCC12CC2 c1(OC)cc(F)ccc1C(=O)NCCCN(C)C(C1(C)CCC12CCC2)=O C(N=S(C)(=O)N(C)C)NCc1cc(N(C)C)ncc1 c1(C(=O)NC(C2(CNC(C3CCCC(O)C3)=O)CC2)C)cccc2c1CC(=O)N2 CC1CC2CC(C(=O)NC(C)CCNC(c3cnc(Cl)c(N)c3)=O)(C2)O1 N1(C(C#C)C)CCN(C(=O)C(C2(O)CCC2)NC(=O)CCc2ccccc2)CC1 C(C(CCCC)NC(=O)CCOCCN(C)C)NC(C1(C#C)CCC1)=O C1(C(N2CCC(CC3CC3)CC2)=O)CCN(C(=O)C2CCc3c[nH]nc32)O1 CN=c1nc(C(N2CC3CC(NC(=O)C=C4CCCC4)CC2C3)=O)cc(C)[nH]1 C1(C(=O)NC2(CN(C(=O)C3=CCCC3(C)C)C)CC2)CCCC12CCOCC2 C1(=CC(=O)NCC(C)(Cn2cccn2)NC(C(C)CO)=O)CCC(C)(C)CC1 CC1(C)CC(C)(NC(C2(NC(=O)CC3CCCNC3=O)CCSC2)=O)C1 c1(C(N2CC(C(C)NC(C3CS(=O)(=O)C3)=O)C2)=O)cc(Cl)c(N)c(Cl)c1 c1(NC(C(C(C)C)N2CCOCC2)=O)c(C(F)(F)F)cccc1Cl c1(-c2ccc(OCC)cc2)ccc(-c2nccn2C(C)CN(C)C)c(F)c1 CC1OC2(C)CC1(C(=O)N(C)CCN(C(=O)C(F)(F)C1CC1)C)C2 Cc1nc2c(o1)CCN(C(c1ncc(Br)cc1F)=O)C2 C1(CCNC(C2CC(F)(F)C2)=O)CN(C(c2cc(C(F)(F)F)ccn2)=O)CCO1 c1(C(N(CCCNC(c2cc(Cl)ns2)=O)CCC)=O)ccc(CC)nc1C C(CN=c1nc2scnc2c(N2CCC(c3cnn[nH]3)C2)[nH]1)c1c(Br)csc1 CC(C)(C)C(C#N)C(=O)NC1CC2CCC1C(NC(=O)COC1CC1)C2 Cn1nc(C(=O)NCC2COC(CNC(=O)CC34COC(C)(C3)C4)C2)cc1Cl C1(C(=O)Nc2c(OC)nsc2)CCCN(C(c2ccncc2)=O)C1 n1(CC)nnc(C(=O)NC(C)(C)C(C)NC(=O)C=Cc2cnc[nH]2)c1C C(=O)(C(CCCOC)NC(c1ncc(F)cn1)=O)NCCn1c(CC)ncc1 C(C)(C)(CC(F)C(=O)N1CC2CC1CN2C)NC(C(c1ccccc1)C)=O N1(C(CCCOCC)=O)CC=C(C(=O)N2CCC2C(C)C)C1 N1(C(C(C2CCC2)OCC)=O)CCCC(C(=O)N(CCC=C(C)C)CC)C1 N(C(=NCCSC)NCCC1CC1(F)F)Cc1ccc(C)nn1 Cc1nccc(CN(C(c2cc(-c3ccccc3)on2)C(=O)NCC(F)F)C)n1 C1(NC(C)=O)CCC(C(N2CC=CC(NC(c3cnn(CCO)c3)=O)C2)=O)CC1 c1(C(=O)NCC2CN(C(CCC=C(C)C)=O)C(C)CC2)c(F)ccc(C#N)c1F C1(NC(C(N)=O)=O)COCCC1NC(c1cccn1C1CC1)=O C1(NC(CSC(C)C)=O)CN(C(=O)CCn2ccc(O)nc2=O)CC1(C)C c1(CC)cccc(CC(=O)NCC2C=CCN2C(c2cnn(CC(C)C)c2)=O)c1 C(C(CC(C)C)NC(=O)C(c1cnn(C)c1)OC)NC(c1ncn(CC)n1)=O C1(CNC(C2C(C)(C)CCCO2)=O)CCC2(CN(C(=O)C(C)(C)S(C)(=O)=O)C2)O1 C(C(=O)Nc1ccc(OC)c(O)c1)(C(C)(C)O)NC(C(CC)=CCCC)=O N1(C(C(CC=C)C)=O)CCN(C(C2CCCOC2)=O)CC12CC2 C(C)(CO)(C(=O)N(CCCN(C(=O)CC(c1c(C)noc1C)C)C)C)OC C1(C(N(CCC)CCNC(=O)COC2(C)CCOCC2)=O)CCC2CC1CO2 N1(C(CC=CCNC(CC2C(C)(C)OCC2)=O)=O)CC2CC1C1CC21 CS(=O)(=O)C1CC(C(N2CCN(C(=O)CNC=O)CC2c2ccccc2)=O)C1 C(=O)(C(O)C(C)C)N1CCC(OCCNC(Cc2ccc(C)s2)=O)C1 C#Cc1ccnc(C(=O)NCC(CC)NC(c2ccon2)=O)c1 N1(C(c2c(C)nco2)=O)CCC2(CCC2)C(CNC(c2cnc(S)n2C)=O)C1 C(=O)(C1=C(Cl)CCOC1)N1CCCC(CC(=O)N(CCc2nn[nH]n2)CC2CC2)C1 c1(C(N2CC(CNC(C(=CC3CCCC3)C)=O)OCC2)=O)cc(C)c(C#N)cn1 CC1C(C)N(C(=O)Cn2cnc(C(F)(F)F)n2)CCN1C(=O)COCC(F)F CC(C(=O)N1CC(NC(c2ccc(CCC(N)=O)cc2)=O)C(C)C1)S(N)(=O)=O C1(NC(C(C)OCCOC)=O)CN(C(c2ccccc2OC)=O)CC12CCC2 CC1CCC(CC(N2CC(C)(NC(=O)Cc3ccn(C)c3)C2)=O)OC1 Cc1ccc(N2N=CC(S(=O)(=O)NCC(N3CCC4(CCCN4)C3)=O)C2=O)cc1 CC1(C)CCC(NC(=O)C(c2cccs2)NC(c2cnc(=N)[nH]c2)=O)C1 CCC(CC(=O)N(C(CC(C)C)C(=O)N(CC(C)OC)C)C)C(C)C C12(C(=O)OC)CC1CCN2C(=O)C(=O)NCc1csc(C#N)c1 c1(C(N2C(CNC(C3(C(C)C)CCC3)=O)CCC2)=O)cc2c[nH]cnc-2n1 C1(N(C(CC(=C)C)=O)CC)CCC(NC(c2ccccc2OC)=O)CC1 c1(CN2CCC(CCNC(c3cc(C(C)(C)C)[nH]n3)=O)CC2)cc(Br)ccc1I C1(C2CCCN(C(c3cc(Cl)cc(Cl)c3)=O)C2)(NC(c2cc(C)oc2)=O)CC1 c1(C(=O)OC)cc(C(=O)N(C2CN(C(=O)C(Cl)=CCl)CC2(C)C)C)c(F)cn1 N1(C(C=Cc2c(OCC)cccc2)=O)CCCN(C(=O)CCC2(C)CC2)CC1C CN(CCc1cn[nH]c1)N1CCC(c2ncc3n2CCCC3)CC1 C1(C2CC2)(CC(=O)N(CCCN(C)C(c2cnco2)=O)C)CC1 C1(C(=O)NC2C(CCC)CN(C(=O)C=Cc3scnc3C)C2)CC2(C1)CC(C)C2 C1(NC(C(F)=C(C)C)=O)CC2CC1N(C(c1c[nH]nc1C)=O)C2 c1(C(=O)NC(C)CNC(c2cc(C3CC3)cs2)=O)ccc(=O)n(CCO)c1 N1(C(CSCCC(C)C)=O)CC(C2CCCN(C(c3ccncc3F)=O)C2)C1 c1(C(N2CCN(c3ccn(C)n3)C3CC23)c2ccccc2)cnc2ncccn12 c1(C(N2CCC(C(=O)NCC(C#C)OC)(C(C)C)C2)=O)cncc(F)c1C c1(-n2cc(C(CCC)NC(c3nc(CCC)sc3)=O)nn2)ccc(F)c(Cl)c1 C(=O)(CCC(=O)N(C(C)CN(C)C(c1cnn(CC)c1Cl)=O)C)NCCC C1(C(=O)Nc2cnc(C)c(Cl)c2)CC2C=CC1N(C(c1cnn(C(C)C)c1)=O)C2 c1(C(C(N2CC(NC(c3nc(CCC)sc3)=O)C2)=O)O)ccccc1C(F)(F)F C1(C(N2CCC(C)N(C(c3nc(Cl)cs3)=O)CC2)=O)CCCC2CCCCC12 C(c1c[nH]c(=N)c(C)c1)=CC(=O)NCC(C1CC1)NC(c1nnn(CC)c1C)=O Cc1c(Cl)ccc(C(C)(C)C(=O)NCC(C)CNC(=O)Cn2cncn2)c1F C(CN=c1ccnc(N2CCC(c3ccco3)C2)[nH]1)(C1CC1)SC Cc1nn(C)c(NC(C2CCCCN2C(c2cnco2)=O)=O)c1C(N)=O C(=O)(C(CC=C)NC(=O)CC(C)C)OCC(N1C(CC#C)CCC1)=O.OC N1(C(c2cn(CC=C)nn2)=O)CCN(C(c2cc3c(s2)CCC3)=O)CC2(CC2)C1 C1(NC(CCCCC)C2CC2)(NC(=O)OC(C)(C)C)CC(C)(C)OC(C)(C)C1 C1(CCNC(Cc2c(OC)nccc2)=O)CCC(C)(C)CN1CCOC N1(C(c2nc(C(C)C)oc2)=O)CC(C)CN(C(=O)CCC2CCCN2C)CC1C C1(C)(CNC(CN(C(=O)C(C)OC(C)(C)C)C(C)C)=O)CC2(CCC2)C1 CC(C)C(F)C(=O)NC(C1CC(N(C)C)C1)C.c12nocc1C(=O)NC2 c1(CC)ccc(C(=O)NC(C)CCCCNC(=O)CC2CCC2C)cc1[N+](=O)[O-] CCC(CCC(=O)NCC1CCCN1C(=O)C1=C(C)CCC1)OC Cc1oc(C#N)cc1C(=O)N(C1CCN(C(c2snc(O)c2Cl)=O)C1)C N1(C(c2c(CC)nco2)=O)CCCC2(NC(=O)C(C)CC(C)(C)C)CCCC12 N1(C(C2(c3ccc(C)cc3)CCC2)=O)CC(CNC(C2CC2(C)C)=O)CC1(C)C C1(CCNC(C(COC)NC(C)=O)=O)CSCCN1C(=O)CC1CCCOC1 c1(C(=O)NCC(CC=C)NC(=O)CCC2CC2(C)C)ccc(C(C)C)nc1C c1(CC(=O)NC2CN(C(c3ccc(F)nc3F)=O)C2)cccc2c1CCC2 C1(OC)(CNC(=O)C(F)n2ccnc2)CN(C(=O)CSCc2cccs2)C1 c1(C(N2C(CNC(C3(C)CCCOC3)=O)CC2)=O)cc(N)c(O)c(F)c1 N1(C(CCC)=O)CCCC1(C(=O)NCCN1CC2CCC2C1)CC C1(C(=O)NC(C)C(c2ccccc2)NC(c2cncc(F)c2)=O)CCN(C)CC1 C#Cc1cccc(CC(=O)NC(C(=O)NCCCCC=C)C2CCCO2)c1 CCCC(CCCNC(c1ccc(-c2ncc[nH]2)nc1)=O)NC(=O)CCCC#N c1(C(=O)NCC2(F)CCCN(C(C3(CC#C)CCC3)=O)C2)cccc2ncsc12 c1(CC)sccc1C(N1CCC(CNC(C2CC(C(F)(F)F)(OC)C2)=O)C1)=O C(C(C)(O)CC(=O)N1CC(NC(=O)C=CCn2cncn2)CC(F)C1)OC CCC(CCCC(=O)N1CCC1C(C)O)NC(=O)C1=C(C)OCC1 c1(OCC(=O)NC2CC(N(C)C(C3CC3C(F)(F)F)=O)C2)ccc(Cl)cc1 c1(C(=O)NC(C)CN(C)C(C23CCCC2C3(F)F)=O)cncc2c(O)nccc12 C1(CC(N2CCC(O)(COC)C2)=O)C2CCCC2N1C(c1cc(C)n(C)n1)=O O=C1OCCCN1CCNC(=O)NC1CC1(F)F c1(OCCCNC(C(=O)N(CC(C(C)C)C)C)=O)cccc(F)c1 c1(OC)nc(C(=O)NCCCNC(=O)C(C)c2ccco2)co1 N1(C(Cc2cc(C(C)C)no2)=O)CCCCC(C2CN(C(C3CC3(F)F)=O)C2)C1 C(=O)(C(C)C(C)(F)F)NCCC1(NC(CC2CC(C(C)=O)C2(C)C)=O)CC1 C1(C(N2CC(CO)C(CO)C2)=O)N(C(C2CCCCO2)=O)CC12CCCC2 Cc1cc(C(=O)NCC2C=CCN2C(=O)C(C)n2cnnn2)c(C)cc1Br c1(C(N(CC(C)NC(C2(Cl)CC2(C)C)=O)C)=O)ccccc1-c1nc[nH]n1 C1(CC(N2CC(NC(Cc3cc(OC)cc(F)c3)=O)C2)=O)COC2(CCC2)CO1 N1(C(c2nc(C)sc2)=O)CC(CNC(c2nnn(C)c2C(F)(F)F)=O)CC1C C1(CNC(CCc2nc(C)c(C)o2)=O)CN(C(=O)CC2CC2(Cl)Cl)CC12CC2 C(=O)(CC1=NNC(=O)C1)N1CCC(C(C)NC(c2cncc(NC)c2)=O)CC1 Cc1cc(C)n(CCNC(=O)CN(C2CCC2)C(C2CC(O)C(F)C2)=O)n1 c1(C(N2CC(n3cc(CCCC(C)=O)nn3)C(C)C2)=O)noc2c1CCCC2 Cc1nc(C(=O)NCCC2=CCN(C(=O)CN(C)CCO)CC2)c2ccccn12 c1(C(N(CC(C)NC(=O)Cc2cc(C)no2)CC)=O)cc2ccncc2cc1F N1(C(C2(OC)CC2)=O)CCOC2(CCCN(C(C3CC=CCC3)=O)C2)C1 CCCC(C(=O)NC1CC(C)N(C(=O)Cn2cnc(=N)[nH]2)C1)OC c1(CO)noc(C2CC2NC2(c3nnnn3CC)CN(C3CC3)C2)n1 S(=O)(=O)(c1nc(N(CC(C)C#N)C)ccc1Br)NCC1(C)ON=C(C)C1 C1(C2CCCCO2)(C(=O)NCc2c(C)nn(CCO)c2)CCCO1 Clc1ccc(CC2(NCc3nccc(I)n3)CCCC2)cn1 Cc1ccccc1CC(=O)N(C1CC1)Cc1ccc(CNC(=O)C=C(Cl)Cl)cc1 N1(C(CCC#C)=O)CCC2(CCCC2NC(c2csc(-c3cnn(C)c3)n2)=O)C1 C#CC1CCCN(C(C2CCC(CNC(C3CCC(CC)CC3)=O)CC2)=O)C1 c1(C(=O)NC2CCC(N(C(c3cnc(CC)s3)=O)C)C2)c(F)c(F)c(F)cc1F N1(C(CCN(C(=O)CC2CC=CCN2C)CC#C)=O)CCCC(F)(F)CC1 C1(n2cc(C(CC(C)C)O)nn2)CCCCC1NC(c1ccn(C2CCC2)n1)=O N1(C(C(C(C)C)NC(c2ccco2)=O)=O)CCC2(C1)CN(C(=O)C1CC1)CC(C)O2 N1(c2cc(C)ncn2)CCC2(NC(c3ccc(F)c(C4CC4)c3)=O)CCCC12 CC(C)(CC(=O)N(CCC(=O)Nc1ccsc1)CCCO)C1CC1 CCCCCCCCCCCC(C)NCCC(n1nc(C)cc1C)OC C1(OC)CN(C(C2(C)COC(=O)C2)=O)CC1NC(c1cc(C)nn1C(F)F)=O CCC(CCOC)C(=O)NCCn1cnc(C(=O)NCCC(CC)CO)c1 C1(OC(F)F)CCCCCC1.C12COC(C1)CNC(=O)C2.C(=O)(CCO)NC Cc1cccc(C=CC(=O)NCCCCC(C)NC(c2cnc(C(C)C)[nH]2)=O)c1 C1(C(N(CCNC(Cc2nc(CC)sc2)=O)CC)=O)CCc2nc[nH]c2C1 c1(C(=O)NCC(CNC(C(CC)C2CCC2)=O)F)cc(Cl)cn1CC c1(SCCC)ccc(C2(C(=O)O)CC2)cc1.C12CCCC(O1)CC(=O)NC2=O C1(C(N2CC(N(c3cc(=O)n(C)cn3)C)C2)=O)CCC2CC2CC1 C1(C(=O)NCCC2(O)CCN(C(C3SCCS3)=O)C2)(OC)CCC(C)(C)C1 CCC(C)C(=O)C(=O)N1CCCCC(C(N2CCCC(C)(CC)C2)=O)C1 c1(N2CC(NC(C3CCC(CC)O3)=O)C(C)C2)nc(C)nc2scc(C)c12 N1(C(C(C2CC2)NC(c2nc(C(C)OC)oc2)=O)=O)CCC(C)(C)CC1 C1(C(F)F)(CNC(C(C)=C(CC)C)=O)CCN(C(c2ccnc(OC)n2)=O)C1 CC1CN(C(C2CCCC3CC23)=O)CC1CNC(=O)C(c1ccccc1)N(C)C N1(C(C(CCC)CC)=O)CC(C)(C)OCC1CNC(c1nccc(Cl)c1F)=O c1(C(N2CCCCC(NC(C(C)N(C)C)=O)C2)=O)cc2cc(F)ccc2o1 c1(C(N(CC(C)NC(C(CC)=CC)=O)C)=O)ccccc1CC(F)(F)F N1(C(C(CC)(C)C)=O)CCC(C2CCCN(C(=O)C(F)(F)c3cscn3)C2)CC1 Cc1[nH]nc(CNC(C2CSCCN2C(=O)CCOC2CC2)=O)c1C c1(OC)ncccc1CNCC1(C(=O)Nc2cc(I)ccn2)COC1 N1(C(c2cccn3nccc23)=O)CCCC2C1CCCN2C(c1cc(Cl)ns1)=O c1(C(C(=O)NCC(C)(CO)NC(C(C)NC(=O)NC)=O)O)ccccc1OC C1(C2CCC2)(C(N(CCCNC(Cc2c(CC)n[nH]c2CC)=O)C)=O)CC1(F)F c1(C(=O)NCC(CCOCC)NC(COCCOCC#C)=O)cncc(C)n1 n1(CC(=O)OC)cc(NC(=O)CC2CCN(CCn3nccc3C)CC2)c(C)n1 Cc1cc(=O)n(C)nc1C(N1CC2(CC(NC(c3coc(CO)c3)=O)CO2)C1)=O c1(OC)ccc(Br)cc1NC(C12CC1CN(Cc1ccc([N+](=O)[O-])s1)C2)=O C1(C)(C(N(CCN(C(C(Cc2c(C)noc2C)C)=O)C)C)=O)CCS(=O)(=O)CC1 N1(C(c2n(C)ccn2)=O)C2CCC1CC(NC(C1CC3(CSC3)C1)=O)C2 C1(OC)CN(C(=O)CC2CC2(Cl)Cl)CC1C(=O)NCCN(C)C c1(OC)cc(CC(=O)NCC2CCC2NC(C23CC(C)(C2)C3)=O)ccc1C C(CCCC(CO)NC(C1C=CC=CC=C1)=O)NC(C(C(C)O)N(C)C)=O N1(CC(=O)C(CCCCC(F)F)=O)CCSc2ccccc21 CCC(CC(=O)N1CCC=CC1COC)NC(=O)C(F)n1ccnc1 CCCCC(O)C(=O)NCCCC1CCCCN1C(c1[nH]nnc1C)=O Cc1cc(C(=O)NCC(C)(CO)NC(c2csc(Cl)n2)=O)nc(O)c1 CCC(C)C(O)C(=O)N1CC(CC(C)NC(C2CC3(CCOC3)C2)=O)C1 C1(NC(C(F)=CC)=O)CCN(C(c2cc(CC)c(CCC)s2)=O)C(C)C1 c1(N(C2CC3CNC2C3)C(C(C)n2cncn2)=O)ccc2cc[nH]c2c1 C=CCC(CNC(=O)C(C)C#N)C(=O)N(CC=C)CC1CC1 c1(CNC(=O)NC(CC)Cc2ccc(Br)cc2)sc2ccccc2c1Br c1(C(=O)NCCOCCOCCNC=O)ccc(P(C)(C)=O)o1.C1(CCOC)CC1 c1(CC)nc(CC(=O)NC2CC(C)(NC(c3n[nH]cc3Cl)=O)C2)cs1 N1(C(C2C(OCC)C2)=O)CCSCC1CCNC(c1cnc(C(F)(F)F)cn1)=O C1(C(N(CCNC(=O)C(C)(C)c2ccns2)CC)=O)Cc2ccccc2C(=O)O1 c1(CC(=O)NC2C(NC(c3c(CC)scc3)=O)CC2)ccc(-n2cnnc2)cc1 C(=O)(C(F)CC(C)(C)C)N1CC(C)N(C(c2cnc(S)n2C)=O)CC1 C1(NC(c2ncc(C)cn2)=O)C(C)CN(C(=O)CCc2ccoc2)CC1C C1(OCCNC(C(n2c(C)ncc2)C)=O)(CNC(=O)C(C)C)CCOCC1 CCC(F)(C(=O)OC)C(=O)N1CCC(NC(=O)COC(C)C)C(F)C1 C1(CCCC)CCC(N(c2nnc(-c3cocn3)n2CCCOC)C)CC1 c1(OCC)nc(C(=O)NCCCCn2cc(CCC3CCCCC3)nn2)ns1 C=C=C(C)CC(=O)N1CCC(O)(CN(C(=O)Cc2cnn(CC)c2)C)C1 CC1CCCC(C)N(C(C2(N=[N+]=[N-])CCN(C(=O)CCn3cccn3)C2)=O)C1 C(=O)(C(C)CC(=O)NC1CCC(C(=O)NCCC(F)(F)F)CC1)OC C1(N(C(=O)Cn2cnnc2O)C)CCCCC1NC(c1ccncc1C(F)F)=O C(=O)(CCCCC(C)(C)C)N1CC(OC)(CNC(=O)CCc2cccc(O)n2)C1 CC(C)(C)CC(=O)NC1CC1CNC(c1c[nH]nc1-c1ccccc1)=O Cc1c(C(N2CCCC2C2CCN(C(c3ccc(NF)cn3)=O)C2)=O)ncn1C N1(C(c2c(C)nn(C(C)C)c2)=O)C2CCC1CN(C(C1CN(C3CCC3)C1)=O)C2 N1(C(Cc2cccc(C(N)=O)c2)=O)CC2COCC(C1)C2NC(=O)C(F)C1CCC1 C1(CC(=O)NC(C)CNC(C2(C(=O)N(c3cnn(C)c3)C)CC2)=O)COC(=O)C1 c1(OC)cccc(C(N2CC3C(NC(C4CCCS(=O)(=O)N4)=O)C3C2)=O)c1OC c1(N2CCC(C(C)O)CC2)ncnc2c1ncn2CCCC1(O)CCOC1 c1(C(N2C(c3ccc(COC)o3)CCC2)=O)ccc2cncn2c1 N1(C(c2cc(COC)no2)=O)CCC(CNC(=O)CC2CCN(C)C2)C12CCC2 C(=O)(CCCS(=O)(=O)N1CCCC1)N1C(C)CN(C(C2OCCOC2C)=O)CC1 c1(C(C(=O)NCCN(CC(C)O)C(c2ccsn2)=O)OC)c(F)cccc1F c1(OCC)cc(C(=O)NC2CCN(C(C3(F)CCOC3)=O)CC2CO)cc(F)c1 c1(CC)nc(C)ccc1NC(C1(C(C)NC(C2CC(C(N)=O)C2)=O)CC1)=O N1(C(C(C)SC)=O)CCC2CN(C(c3c[nH]c(C(C)(C)C)c3)=O)CCC12 Cc1nnc2n1CC(C(=O)NCC1CC1NC(c1nnn(C(C)(C)C)n1)=O)CC2 CC(C)(CCCF)NC(=O)C(C)(CO)NC(c1cnc(Cl)s1)=O c1(C(N2CC3C(NC(C(COC)CC(C)C)=O)C3C2)=O)cn(C)c(C)c(Br)c1=O CC1(C)C(NC(=O)C(N)=O)CCN1C(=O)CC(=O)NCC1CC1 Nc1cccc(F)c1OCCCCC1CCCOC1 c1(C(=O)Nc2c(C)ccc(Br)n2)nc(C2=CCC(C)CC2)cs1 Cc1ncc(F)c(=NCC2CCCCN(C(=O)CC(C)(O)C3CC3)C2)[nH]1 C1(F)(CNC(c2cc(C)n(CCO)n2)=O)CCCN(C(c2cnc[nH]2)=O)C1 c1(C(N2CC(Cc3ccn(C)n3)CC(F)(F)C2)=O)ccc2c(n1)NC(=O)CC2 Cc1cnc(C(N2CCC(C)C2CNC(=O)Cc2cccc(F)c2)=O)cc1Cl c1(C(=O)NCCCC(C)NC(CCc2cc(C)no2)=O)cc2c(s1)CCCC2 C1(C)(C(=O)NCCc2c(CNC(CC3(CSC)CC3)=O)nco2)CC(C)(C)C1 Cc1cc(NC(=O)CCC2CCCN2C(C2CCN(C)C2)=O)cc(C)c1Br C12(C(N(C3CCCC3)CC=C)=O)CCC1CN(C(=O)C1=C(C)OCC1)C2 C1(C(=O)NC(C(=O)N(CC(F)(F)CO)C)CCC2CC2)CC2(C1)CC21CC1 N1(C(c2ccc(CC)[nH]2)=O)CCCC(C)(C)C1CNC(=O)CC1SC(=N)NC1=O CCC(CC(=O)N1CCCC(N(CCF)C(=O)NC2CCC2)C1)CC(C)C O=C(CCCCCCCCC1CC1)NCCNC(c1cnc2c[nH]nc2c1)=O N1(C(c2c(CC)scc2)=O)CC(NC(=O)C(C)NC(C)=O)C2(CC2)C1 N1(C(CN2CCN(CC)CC2)=O)CCCC(NC(C2(C(F)(F)F)CC2)=O)C1C CCC(C(=O)N(C1CCN(C(=O)Cc2ccon2)C1)Cc1ccccc1)C(C)C c1(OC)nsc(C(=O)NCC2C=CCN2C(=O)C=CC(F)(F)F)c1Br CC1CN(C(=O)CC2CC3(CCC3)CO2)CCCN1C(c1ccccc1Br)=O Cc1[nH]nc2c(C(=O)NCC(C3(O)CCN(C(c4cncs4)=O)C3)C)cccc12 C1(C(=O)NCCOCCC(=O)NC(C(N)=O)C2CC2)(CO)CCCCC1 C(=O)(C1=CCS(=O)(=O)C1)NCCC1(NC(CC2C(C)CCO2)=O)CCCC1 c1(C(N2CCCC(c3nncs3)C2)=O)cn(CCC(F)(F)F)nc1-c1ccccc1 CC1(C)CCN(N2CCCC2COc2ccc(F)cc2F)CC1 N1(C(C2CC(CC)C2)=O)CCC(c2nnc(CNC(C3CC3F)=O)s2)CC1 c1(C(=O)Nc2cccc(C)c2F)ccc2ccc(O)cc2c1 C1(N(C(C(C)OCC=C)=O)CCO)CCCN(C(c2nc[nH]c2C(C)(C)C)=O)C1 c1(C(N2C(C(=O)NCC(C)OC)CC(F)(F)C2)=O)cc(I)c(F)cc1F c1(C(=O)NCCn2cc(C(N(CC(CC)C)C)=O)nn2)ccc(C)cc1C C1(N(C)C)CCC(C(N2CC(=C(F)CNC(=O)C(O)CN3CCCC3)C2)=O)CC1 C(=O)(C(CCC1CC1)NC(c1sc(C)cc1C)=O)N(CC(=O)N(CC)CC)C N1(C(C2C(CCC)CCC2)=O)CCN(C(c2cnn(C(C)(C)C)c2N)=O)CC1C C1(C(=O)Nc2cccnc2)(CC)CCN(C(c2cccc(CO)c2)=O)C1 N1(C(C2CN(C(C)=O)C2)=O)CC2CCOCC2(NC(c2ccc(C)s2)=O)C1 C(=O)(C1=CCC(NC(=O)C(C)n2cccc2)C1)NC(C(=O)OC)C1(C)CC1 N1(C(=O)C=Cc2ccco2)CC2(CCCC2)C1C(N1CCC2(CCC2)CC1)=O N1(C(Cc2n(C)nnc2)=O)CCC2CCC(NC(C3CCCC(C)(C)C3)=O)C1C2 Cc1cc(C(N)=O)cc(C(=O)NC2(CCNC(c3cscc3C(F)F)=O)CC2)c1 C1(NC(COc2cc(C)on2)=O)CCN(C(=O)C=C2CN3CCC2CC3)CC1F C(CCC(O)CO)N(C)C(C1(CNC(=O)CC2OCCCO2)CC=CC1)=O N1(C(C(CCCC)NC(C2C=C(C)CS2)=O)=O)CCC(O)C(C)(O)C1 C1(NC(CCC#C)=O)(CNC(=O)C(c2ccncc2C)C)CCCCC1 c1(C(=O)NCC(C2CCOC2)NC(c2ccc(OC)o2)=O)nc(C)ccc1C c1(C(C)CC2CCN(C(N=c3ncn(CC)[nH]3)=O)CC2)cccc2nn(C)cc12 C1(C(=O)NC2CN(C(c3cnnn3C3CC3)=O)CCC2O)CCn2cnnc2C1 C(=O)(C(C)(C)NC(=O)OC(C)(C)C)NC(CC)CN(C)C(c1cnsn1)=O c1(NC(C2N(C(C3CC=C(C)CC3)=O)C3C(C2)C3)=O)cc(Cl)c(O)c(Cl)c1 n1(C(C)C)cc(C(=O)NC2CCC(CNC(=O)CC3CN(C)C3)C2)c(O)nc1=O c1(NC(C2(n3cc(CCC(CC)O)nn3)CC2)=O)ccnc2cc(Cl)ccc12 C12(NC(C(C)OCCC(C)C)=O)CCCN(C(c3c[nH]c(=O)cn3)=O)CC1C2 C1(O)(CC)CCCN(N(C(=O)CCn2cnnn2)C2CN(c3ncccn3)C2)C1 C(=O)(C1=CCC(C)(C)CC1)NC(CCCOC)C(=O)NC(C)CSC C(=O)(C#CC1CCOCC1)Sc1c(NC(=O)CCCSc2ccccc2)ccs1 C=CCCC(F)(F)C(=O)N(CC(O)CN(C)C(c1ccnc(SCC)c1)=O)C C12(C(N3CCC(NC(c4c(F)ccc(F)c4Cl)=O)C3)=O)CCC(F)(CC1)CC2 C(C(=O)NCC(C)N(CCSC)CC)NCCC N1(C(c2c(OC)n[nH]c2)=O)C(CNC(C2CC(C)(C)CO2)=O)CC2CCCC12 c1(C(=O)Nc2cccc(O)c2)cn2c(n1)CN(Cc1ccc3ccsc3c1)CC2 C12(C(=O)NC3CCC(NC(=O)CCc4cccnc4)CC3)CSCC1C2(F)F c1(C(N(C)CC2CCN(C(C3CC4CC34)=O)CC2)=O)ccccc1[N+](=O)[O-] c1(C(=O)NC(CNC(c2cn(CCC)nc2)=O)C)nccn2c(C)nnc12 c1(CNC(C(n2ncc(C)c2)C)=O)ccc(CNC(=O)C=Cc2ncc[nH]2)cc1 C1(NC(C=CSC)=O)CCS(=O)(=O)C12CN(C(c1nc(C)ccc1C)=O)C2 C1(C(=O)NCCOC2CN(C(C3C(C)CC(=O)N3)=O)C2)C2CCC(C2)C1(C)C Cc1nccc(CN(C(=O)CCCn2cc(C(C)O)nn2)C)n1 c1(C(N2C(C3C(=O)NCC3)CCC2)=O)ccncc1-n1cccn1 CC1(CCNC(C2CC2F)=O)CCN(C(c2ccc(F)cc2N)=O)CC1 c1(C(=O)NC2C(NC(CSCCCC)=O)C2)ccc(C(=O)N(C)C)nc1C c1(C(=O)NC(C)C)ccc(C(=O)NCC2C=CCN2C(c2csnc2Cl)=O)cc1 Cc1cncc(C(N2CC(=O)CC2C(N2CCC(CC(F)F)C2)=O)=O)n1 Cc1noc(C)c1S(=O)(=O)NC1CCN(Cc2n[nH]c3ccccc23)CC1(C)C CC1CN(C(=O)CNC(=O)C(C)(C)C)CC1(C)CNC(=O)CSS(C)(=O)=O c1(C(=O)NCC2(COC)CCN(C(=O)COC(C)=O)CC2)cc2cnccc2[nH]1 Cc1cc(CC(=O)NCC2CCN2C(=O)C(C)(F)F)sn1 C1(N(C(=O)C=C(Cl)Cl)C)CC2CCC(C1)N2C(=O)CSC1CCOC1=O c1(C(=O)NCC2OCC(CNC(c3csnn3)=O)C2)ncc(Cl)cc1Cl c1(CNC(C(C(CC)CC)OC)=O)ccc2c(c1)CN(C(=O)C(C)(C)OC)C2 c1(CC)cc(C(N2CCC(F)C(NC(=O)COCc3nc[nH]n3)C2)=O)ccc1Cl N1(C(C(CC)OCC)=O)CC(C)(C(=O)NCc2ccncn2)CC1(C)C N1(C(C=CCCC(C)C)=O)CC(C)N(C(=O)C#CC2CCOC2)CC1C C#CC1(NC(C2(C#N)CC23CCC3)=O)CC2(CCOCC2)C1 Cc1[nH]c(C#N)cc1C(=O)NC1C2CC(NC(C3CC3C3CCC3)=O)CC12 N(C1COc2ccc(Br)cc21)C(=O)OCCc1cccc(OC2CCCCC2)c1 C(C)(C(=O)NCCN(C(=O)C(C)C1CCOC1)C(C)C)OCCC=C C1(C(C)C)C(CO)CN1C(=O)CCOC1CN(C(=O)C=CCN2CCCC2)C1 CCCC(C)CC(=O)N1CC(NC(C2(C#N)CCOCC2)=O)CC1(C)C C(=O)(C1=NOC2COCC12)N1CC2C(NC(c3c(N(C)C)nccc3)=O)C2C1 CC(C)(O)CC(=O)NCCOC1CCN(C(c2cccc(C(N)=O)n2)=O)C1 C1(CC)CC(C(N2CC3CC2C3CNC(=O)CSC(C)C)=O)CC(=O)N1 N1(C(COC(C)C)=O)CCC(CNC(C2CCCNS2(=O)=O)=O)C1(C)C CC(C)CCC(O)C(=O)NC1COCCC1C(N1CC2(CCOCC2)C1)=O C1(C(=O)NC(c2cn(C(COC)C)nn2)CC(N)=O)(OC)CCOCC1 c1(OCC(N2CC(O)CC(NC(c3c(C)noc3N)=O)C2)=O)nc2ccccc2s1 N1(C(c2c(C(C)C)noc2)=O)CCC(NC(=O)CCN2CCC2)CC(C)(C)C1 c1(C(=O)NC2(CNC(C=Cc3ncc(C)[nH]3)=O)CCCC2)nc2cnccc2s1 C1(OC)C(OC)CN(C(=O)C2=CCCC2)C1CNC(=O)Cc1csc(Cl)c1 CC(C)C(F)(CNC(C1CCCO1)=O)C(=O)N1CC(N(C)C)C1 CC1CCc2c(C(=O)N(CC(O)CNC(=O)C#CC3(C)CC3)C)csc2C1 CCCC(C)CC(=O)N(CC(=O)NC(CCNC(N)=O)=O)CC C1(C(=O)NCC2CC(F)CN2C(c2cncs2)=O)CC2(C1)CC(F)C2 C#CC(CNC(C1(CC)CN(C(=O)Cc2ccc[nH]2)C1)=O)C(C)C CCCC(C)CC(=O)NCC12CC(NC(C3CC3c3ccnn3C)=O)(CCO1)C2 N1(CC(=O)NC2(C3CCCN3C(=O)Cc3cccc(F)c3)CC2)CC2CCC1C2 C1(C(=O)NC2CCC(C)N(C(=O)C(C)(C)F)C2)CCc2ccnn2C1 Cc1cc(N2CCC(Cc3cccc(F)c3)C2)nc(=NCCc2ncc[nH]2)[nH]1 N1(C(C2CC3(CC(=C)C3)C2)=O)CC2CCCC(CNC(=O)C(C)(O)CCC)(C2)C1 C12(CCOCC1)CS(=O)(=O)NCCO2.C(=O)(CC(F)(F)F)OC c1(OC(C)C)nc(N2CCN(C(=O)Cn3ccnn3)C(CC#N)C2)ncc1Br C1(NC(C2CC(C)N2C(c2ccccc2C#N)=O)=O)CC2(CCCC2)C1 C(C(=O)NC1C=CCN(C(C2CC(C#N)C2)=O)C1)(C(C)(C)C)NC(=O)OC(C)(C)C c1(C(N2CCC(NC(c3c(CCC)n(CC)nn3)=O)CC2)=O)cc(F)ccc1O N1(C(C2C(=O)NC(=O)N2)=O)CCC(C2(NC(=O)C(C3CCCCC3)F)CC2)CC1 Cc1cc(CCNC(C23CC(NC(=O)CC4COCCO4)(C2)C3)=O)on1 C1(C(N2CCC(C(CC)C)CC2)=O)CCN(C(c2csnc2OC)=O)C1(C)C C(=O)(CCC(=O)NCC1(CCCC)CCCC1)NC1C(C(=O)OC(C)=O)CC1 c1(C(N2CCC(NC(=O)CSc3nc[nH]n3)CC2)=O)c[nH]c2cc(Br)ccc12 c1(-n2cc(C(CC(N)=O)NC(c3ccc(Cl)cc3)=O)nn2)ccccc1C(=O)O C1(CNC(C(C)=C2CCC2)=O)C(C)CCCN1C(=O)CN1CCN(C(C)C)CC1 N1(C(CCc2onc(C)n2)=O)CC(NC(=O)C2=NOCC2)CC1C C1(NC(=O)CCC2CCCCC2)CCCCC1CNC(c1nsnc1O)=O c1(C(=O)NCC(CC)(CC)NC(C2CCNC2=O)=O)cnc(SC)nc1O Cc1cc(=NC(=O)C2CCN(C(=O)CC3CCC(=O)CC3)CC2O)[nH]n1C(C)C C(=O)(CCCCC(C)(C)OC)N1CCN(C(C2CC(CC)(CC)C2)=O)CC1CO C1(C)(C(=O)NC(C)CCCNC(c2c[nH]c(C(F)(F)F)c2)=O)CCC(C)C1(C)C C12(C(N3CC4C(CO)C4C3)=O)CC3CC(CC(C3)C1)C2 C12(CNC(c3nccc(C(F)F)n3)=O)CC(CO1)N(C(c1csc(F)c1)=O)C2 Cc1cc(F)cnc1C(N1CCC(F)(C(=O)NCCC(C)N2CCC2)C1)=O CC1CN(C(=O)CC2CN(C(c3cncnc3)=O)C(C)(C)C2)CC(C)(C)O1 c1(C(=O)OC)ncccc1NC(c1cc(NCc2cccc(OC)c2)cn1C)=O CCC1=C(C(=O)NC(C)C(C)NC(=O)Cc2ccc(O)cc2)CCCO1 c1(C(N2C(C(=O)Nc3ccc(C)c(I)c3)CCC2)=O)ccc(C#N)cc1F c1(C(=O)NC(C(=O)NCCS(CC)=O)C(C)C)ccc2[nH]ccc2n1 c1(C(c2n(CCSC)nnn2)NCc2ccsc2Cl)nc(Br)ccc1C C1(CC(=O)NC2CC(C(C)NC(c3cccn3C)=O)C2)CCCC(=O)C1 O(NC(=O)C1=CCC(NC(C2CCC(C#N)CC2)=O)C1)CCOC C1(C(C)NC(CCNC(CCCOC)=O)=O)CN(C)CCO1 C1(NC(COCCC=C)=O)CC2(CCN(C(c3c[nH]nc3C(F)F)=O)CC2)C1 C1(NC(C#C)CC(C)C)CCC2(CCCNC2)C1 Cc1cnccc1C(N1CCC(C(C)NC(=O)C=CCF)C1)=O c1(CC)onc(C(N2CCC(C(N3CCC(CF)C3)=O)CC2)=O)c1C c1(C(N2CC(CNC(C3(C)CC=CC3)=O)C2)=O)cncc(F)n1 c1(SC)ncc(C(=O)NCCNC(C23CCCC2(C(N)=O)C3)=O)c(O)n1 CCCC(C(=O)NCCC1CC(NC(=O)C(C)NC(=O)CC)C1)NC(C)=O N1(C(C2CCC(CC)O2)=O)CC2(CCN(C(c3cnc(C4CC4)[nH]3)=O)C2)C1 c1(SCC)cc(C(=O)N(C)CC2COCCN2C(=O)CCC2CCCO2)ccn1 CCC(C)(CC(=O)NCC(=O)NCc1cn(-c2cccnc2Cl)nn1)OC(C)=O C1(C(=O)NC2CCC(N(C)C(C3CC4C=CC3O4)=O)CC2)CCC2(CC1)CC2 c1(C(C(=O)NCCSC)N(c2ccc(F)cc2)CC)cnc2c(F)cccc2c1 N1(C(C2N(C(CC)=O)CSC2)=O)C2CCC1C(CNC(c1sccc1F)=O)C2 CC12CN(C(=O)CNS(=O)(=O)c3ccccc3)CC1CN(C(C1C=CCC1)=O)C2 c1(CN(C(C2C(NC(C(CC)C)=O)CCO2)=O)C)ccccc1C c1(OC)cc(C(N2CC3CN(C(C4(C)CCCCC4)=O)C3C2)=O)ccc1C N1(C(CN(C(CCOCCCOC)=O)CC2CC2)=O)CC(=O)N(C)CC1C c1(C(=O)NC2CN(CC)C2)cccc(CNC(=O)C(c2cccnc2)N)c1 C1(COC)CN(C(C2CC3(CC3)CO2)=O)CCN1C(c1coc(C(F)F)c1)=O c1(OC)ccc(C(=O)NCCC2CCCN2C(C2CC(O)C2)=O)c(OC)c1 C#CCCCCCC(=O)NC1(CO)CCCN(C(c2ccccc2COC)=O)C1 CS(=O)(=O)c1ccc(C(=O)NCC2CCN(C(c3cccnc3)=O)CC2(F)F)[nH]1 CN1C(=O)CC(C(=O)NCC(O)CNC(=O)C(C)(C)C(N)=O)C1c1ccnn1C C(CCCC(=O)NCC1(NC(=O)CCCC2CC2)CCOC1)OCC C(CC1=CCCCC1)NC(C1(CNC(c2c(COC)cc[nH]2)=O)CC12CCC2)=O CCC(O)C(C)(C)C(=O)NC(CNC(c1ccc(CO)nc1)=O)C1CCC1 Cc1cc(C)c(NC(=O)C(c2ccns2)N(C)C(C2CCC2)C)c(C)c1 Cc1noc(C(=O)NC(C2CCN(C(c3c[nH]cc3Br)=O)CC2)C)c1C C1(C(N(C2C(CC)CCCC2)C)=O)CCN(C(c2ccc(F)cc2F)=O)CC1C N1(C(=O)NCc2ccc(C)cc2)CCC(CNCc2ccc(Br)c(C)n2)C(F)C1 C1(C)(CNC(=O)NCC(C2CCCOC2)OC)CC2(CCC2)C1 c1(CCCNC(=O)NC(c2ccncc2)CC2CC2(C)C)cc(C(F)(F)F)n[nH]1 CC1(C)CCCC(C(=O)NCC2(C)CCN(C(=O)CCCc3ccccn3)C2)C1 Cc1cnc2c(C(=O)N=c3ccn(C(F)(F)F)[nH]3)c(Cl)ccc2c1.N1CCCC1 CC1CCCC1C(=O)NCc1cc[nH]c1C(=O)NCc1nc[nH]n1 C1(CC)C(=O)N(C)CCN1C(C1(C(C)NC(=O)C(C)CC2CC2)CC1)=O C(C(C)CC(=O)NC1(C(=O)NCCCCCSC)CC1(C)C)OC Cc1cccc(-c2nc(CC3CCCCN3Cc3cc(Cl)c[nH]3)cs2)n1 c1(SCC)ccc(CC(=O)NCC2CC(O)(CNC(=O)C(O)CC)C2)cc1 C(N=c1cc(NCCC(C)CO)nc(C)[nH]1)c1cccc(OC)c1C C=CC(C)(CCOC)C(=O)NC(C)CC1CN(C(=O)CCc2cn[nH]c2)C1 N1(Cc2c(OC)ccc(OC)c2)CCC(NC(c2nocc2C)=O)C(C)(C)C1 Cc1ccc(C(=O)NCC(=O)NCCC2CC(NC(C34CC(F)C3C4)=O)C2)cc1 C1(N=[N+]=[N-])(C(=O)NC(CN(CCCC)C)C)CCN(C(=O)CC2C=CCCC2)C1 c1(OC)ccc(C)c(C(=O)NCC2(NC(=O)Cn3cnnc3C)CC2)n1 CC(C)CC(C(=O)N(C)C)ONC(c1cccc(C2CC2)c1F)=O c1(C(N2CCCC(C)C2CCNC(C2(F)CC2)=O)=O)cccc2c1COCCN2 N1(C(C(C)(C)F)=O)CCC(CNC(C2CC(C)(C)CO2)=O)C(F)(F)CC1 C1(N(C)C(c2nocc2Cl)=O)CN(C(c2ccc(Br)o2)=O)CC12CC2 Cc1nn(C)c(Cl)c1C(=O)NCC(C1CCN(C(=O)C=CC2CC2)C1)(C)O c1(C(N2CC(CC(C)NC(Cc3scc(C)c3)=O)C2)=O)cnc2cccnc2c1 O=S(=O)(c1cccc(N2CCN(c3ccncn3)CC2)n1)Nc1ccnc(Br)c1 C1(NC(=O)COCC2(F)CC2)CC12CC(NC(c1n[nH]c(C3CC3)c1Cl)=O)C2 C1(O)(CNC(C2CSCCN2C(=O)Cn2nccn2)=O)CC2C=CC1C2 C1(NC(C2N(CC(C)C)CCC2)=O)CN(c2ccnc(C#N)n2)CCC1C N1(C(CC)=O)CCCC(C(N2CCC(N(C(=O)CCc3nc[nH]n3)C)C2)=O)C1 C(=O)(C1=CCC2(COC2)OC1)N1CCC(C)(NC(c2nn(C)c(F)c2)=O)CC1 c1(C(N(CCc2cn(C(C)C(=O)O)nn2)C)=O)ccc(Br)c2cn[nH]c12 c1(C(N(C2CN(C(=O)COCCF)CC2(C)C)C)=O)cc2cnccc2o1 N1(C(Cn2cc(C(C)=O)nn2)=O)CC2CC(NC(=O)CC3CN(C)C3)C1C2 c1(C(N2CCC(CC(=O)NOCC(F)(F)F)CC2)=O)ccn2ccccc12 Cc1cc(Cn2cc(C3CCN(C(=O)CCCC(C)C)C34CC4)nn2)ncc1F C(CCN(C(=O)CC(C)(C)O)C)(C(C)C)NC(CCN(CCCCC)CC)=O C=CC1COCC1COC(=O)C(CCOC(C)(C)C)N(C)C C#CCCCC(C)C(=O)NCC1CC(C)(C)CN1C(c1ccnc(OC)c1)=O N#Cc1cc(S(=O)(=O)N2CC3CC2C3C(=O)Nc2cc(F)ncc2F)ccc1Br C1(C(=O)NCCOCCC(=O)NCC(C)(C)n2cccn2)CCCCO1 CC(C)CC(C(=O)NCc1ocnc1C(=O)NCC(C)(C)CCCO)C(N)=O c1(C(N2CC(O)(C(C)NC(=O)CNC(N)=O)C2)=O)ncc[nH]c1=O C(CCCC)(C(=O)Nc1cccc(OCF)c1)NC(C(C=C)OC)=O c1(C(=O)NC23C(CN(C(C(CC)n4cccn4)=O)C2)C3)cc2[nH]nc(C)c2cn1 CCC(CC(=O)N(CC(C)C(=O)N(C)Cc1cccc(O)c1)C)SC c1(C(=O)NC2CCC(NC(c3c(C)ccc(F)c3)=O)CC2)cnc2cccnn12 c1(OC)cc(C(=O)NC2(C)CCN(C(C3CCO3)=O)CC2)sc1S(N)(=O)=O CCC(F)(F)CC(=O)N(C)CC=CC(=O)NC(C)CS(C)=O C1(CNC(=O)C=CC2CC2)CN(C(c2cnc(N3CCCCC3)s2)=O)CC1O c1(NC(=O)C=CCC2(NC(=O)CN3CCOCC3)CCC2)ccc2ncnn2c1 N=c1ncc(C(=O)NC2CCOC(CNC(C3CC(OC(C)(C)C)C3)=O)C2)c[nH]1 c1(CCC(=O)NCC(C2CCC2)NC(CC(C)n2cccn2)=O)ccc(Cl)nc1 c1(C2(C(=O)NC(CNC(C3(CC)CCOCC3)=O)CO)CC2)ccc(F)c(F)c1 C1(NC(C(n2c(C)ncc2)C)=O)CC2(C1)CN(C(c1ccccc1C1CC1)=O)C2 c1(C(c2n(CCCC)nnn2)NC(=O)CCCOC(C)=O)cc(NC(C)=O)sc1C c1(CC(=O)NC(COCCOC)Cc2ccccc2)ccc(OC(C)C)cc1 c1(OC)ccc(CCCC(=O)NC2CCCN(C(=O)Cn3ccnc3C)C2)cc1 c1(OC)ccc2c(c1)C(n1cc(CNc3nccc(CC#N)n3)nn1)CCO2 c1(OCCC)ccc(C(=O)NC2C3CN(C(C4CCCN4C(N)=O)=O)CC23)cc1 C(=O)(C(CC)C(C)O)N(CC1CCC(N(C(CCOCC#C)=O)C)CC1)CC CCC(CC)CCC(=O)N1CCC(CNC(C2CSC2)=O)C(O)C1 c1(NC(C(C)N(C)C(C2CC3CC3C2)=O)=O)ccc(N2CCOCC2)cc1 c1(-c2cccc(OCCC)c2F)c[nH]c2cc(C(=O)NCCCCCO)ccc12 C1(NC(=O)CC2(N3CSCC3=O)CC2)CN(C(=O)CCCn2ccnc2)CC1O c1(NC(=O)NCC2CN(C(c3c(C(=O)OCC)[nH]cn3)=O)C2)ccc(F)c(Br)c1 N1(C(c2cnc(C(C)C)[nH]2)=O)CCCCCC(NC(C2CCCOCC2)=O)C1 C1(C)(C(=O)OC)CC(F)CN1C(=O)C(C)C=C(C)C CN1CCN(C(=O)CCC2(C)N=N2)CC1C(=O)NC1C=CCCCC1 C(C(C)CN=c1[nH]c2c(c(=NC(C)c3ccncn3)[nH]1)CCC2)OCC c1(OC)ccc(C)nc1C(=O)NC(C1CCOC1)CNC(=O)CC=CC(C)(C)C c1(C(C)(C)OC)cc(C(=O)N(C)CCOC2CC3(C2)CC3F)cc(O)n1 n1(CCSC)nnnc1C(c1cc(C2CCC2)[nH]n1)NCc1ccno1 C(CCCC(CO)NC(c1ccnn1C1CC1(F)F)=O)NC(=O)CC1CSC1 N1(C(=O)Nc2c(SC)cc(F)cc2)CC2CC(C1)CS(=O)C2 Cc1nc(C)c(CNC(C2(C)CCN(C(C3CC(O)C(F)C3)=O)C2)=O)[nH]1 c1(N2C(CO)CC(C)(C)C2)nc(=NCc2ccc(CO)o2)[nH]c2cc[nH]c12 CC1C(C(=O)N2CC=CC2C(N2CCCC(CF)C2)=O)=NOC1C N1(C(CCSCCCC)=O)CC(NC(c2sccc2SC)=O)CCC1C n1(CC)cc(Br)c(SNC(CN2CCN(CCC3CC(=O)N(C(C)C)C3)CC2)=O)n1 C1(NC(C(CN(C)C)N(C)C)=O)CCCCC1NC(=O)COCCn1cncn1 c1(C(N2CC(NC(CC(C)(C)C)=O)C(c3ccccc3)C2)=O)nccc(Cl)c1F C1(C(=O)NCC(CC)NC(c2cc(C(N)=O)c[nH]2)=O)Cc2ccc(F)cc2O1 c1(CS(=O)(=O)NCC(c2c(OC)cccc2)O)cc(Cl)c(Br)c(Cl)c1 N1(C(c2csc(CO)n2)=O)CC2(C1)CN(C(C1CC1[N+](=O)[O-])=O)C2 CN=c1nc(C(=O)NCCC(C)N(C)C(c2csc(C(C)(C)C)n2)=O)cc(C)[nH]1 c1(C(N(C(C)CCNC(C2CC(CCF)C2)=O)C)=O)ccc2c(c1)C(=O)NCC2 C1(C)(NC(C(c2cc(C)sc2)(F)F)=O)CCN(C(C2(O)CCOC2)=O)CC1 CCCCC(CC)C(=O)NCCCNC(c1cc(N2CCNC(=O)C2)ccn1)=O CC1(C)CN(C(c2ccoc2Cl)=O)CCC1NC(=O)CC1SC(=N)NC1=O CC(=O)CCCC(=O)N(CCCNC(=O)CC1CCC(C)(C)CO1)CCO C1(C(=O)NCC(CC)NC(c2cccc(CCO)c2)=O)(CO)CC(F)(F)C1 N(C1CCCN(C)c2ccccc21)C(CC(CC)(C)C(=O)OC)=O n1(CC)cc(CC(=O)NCC(CNC(=O)Cc2cncnc2)CO)c(C)n1 C1(C#N)(C(=O)NC2CC(C)(CNC(CNC(=O)NC)=O)C2)CC2(CCC2)C1 c1(-c2cn(CCN(C(=O)CCc3cncn3C)CCOC)nn2)cnn(C)c1C C1(C(=O)NCCOCC(=O)NC(COC)C)CC(SC)C1 C1(CCNC(C2CC2F)=O)CC(N=c2[nH]c(Cl)ncc2F)C1 N1(C(c2ccn(CC)n2)=O)CC(CNC(=O)C=Cc2ccc(C)o2)N2CCC1C2 c1(C(=O)NCC(CC)NC(c2scnc2C(F)F)=O)cccnc1COC c1(C2CS2)ccc(Cl)cc1.n1(C2(NCC(=O)OCC)CC2)cccn1 N1(C(CNC(=N)N)=O)CCC2C(CCN2C(c2ccccn2)=O)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CC(Cn2cc(C(C)(C)OC)nn2)C1 C12(NC(=O)COCCF)CCCC1N(C(c1ccoc1C(F)(F)F)=O)CC2 C(C)(C(C)(C)C(=O)NCC(C)N(C)C)NC(COCC(=O)NC)=O C1(CNC(c2c(C)nc(CCC)o2)=O)CC2CCC1N(C(C1CCC3CC13)=O)C2 C=CC1CN(C(=O)C(F)(F)c2cnn(C)c2)CC1NC(c1cccs1)=O Cc1cc(N)c(C(N2CC(C3CN(C(=O)C(C)N(C)C)C3)C2)=O)c(F)c1 C1(C(=O)NCC(C#C)CC2CC2)CN(C)CCN1C(=O)CC(C)(C)CN(C)C c1(CC(N2CC(NC(C(CCC)OCC)=O)C2)=O)c(Cl)ccc(O)c1Cl C1(CNC(c2c(C)nc(C)s2)=O)COCCN(C(C2CC(=O)C2C(C)(C)C)=O)C1 C(=O)(CC(=O)NC(Cc1cnc[nH]1)C(=O)NCC(C)(O)C1CCC1)OC Cc1ccc(CNC(=O)COC2CCN(C(=O)C(Cl)Cl)C2)cn1 c1(CCNC(N)=O)ccc(C(=O)NC(CC2=NOCC2)=O)cc1 C(=O)(CCCCC(C)(C)C)NCC(CC)(C)NC(=O)Cc1ncn2c1CCC2 c1(C(=O)NC2CCN(c3ccnc(C(C)C)n3)C2)cc[nH]c2nccc1-2 c1(CN2CC(F)CC(C(N3CCS(=O)CC3)=O)C2)ccc2ncnn2c1 Cc1ccccc1C1CCN(C(=O)NCc2ccccc2O)C1.c1(S)nccn1C C(=O)(C1=CCCOC1)N1C(C(=O)NCC(=C)F)CC1C C1(C(=O)NC(CC#C)C(N)=O)CN(C(C2CCC(C(=O)OC)O2)=O)CC(C)O1 C1(CNC(=O)CSC2CCOC2=O)COCCN1C(=O)Cn1cccc1 C1(CNC(C(C)C(F)F)=O)CC(F)(F)CN1C(=O)COCc1ncnn1C N1(C(C2CC3C=CC2C3)=O)CC2(CCN2C(c2cccnc2S)=O)C1 c1(OC)cc(CC(N2CCC(NC(C3CC(Cl)(Cl)C3)=O)C2(C)C)=O)ccc1F Cc1cnc(C(N2CCC(NC(=O)CC3CCCC(C)O3)C2)=O)cc1C#N N1(C(CCCOC)C(=O)Nc2ccc(OC)cc2C)CCCCC2CCCCC12 CN1CCCC(F)(C(=O)NCCC2CN(C(=O)Cc3csc(=N)[nH]3)CCO2)C1 c1(Cc2cc(C(N(CCNC(C3CC(CC)C3)=O)CC)=O)on2)cccc(Cl)c1 N1(C(C2C(C)CCO2)=O)CC(NC(C2(C#N)CC(=O)C2)=O)CC1C Cc1cccc(OCCN(CCCN2CCOCC2CC(O)C2CC2)C)c1 c1(C(N(C)CC2(NC(C3C(C)CCC3)=O)CC2)=O)ccnc(OC2CC2)c1 Nc1c(C(N2CCCC2CNC(=O)CSCc2ccccc2Cl)=O)cccc1F CC1OC2(C(=O)NCC3CC(O)CN3C(C3CC3C(C)(C)C)=O)CCC1CC2 C1(NC(C2C(NC(=O)CCn3cccn3)CCC2)=O)CCCCCC1 Cc1cc(Cl)c(S(=O)(=O)NC2CCC(F)(F)C(C)C2)c(Br)c1 C1(NC(CCC=C(C)C)=O)(CNC(=O)CCn2ccnc2C)CC2CCC1CC2 c1(C(N2CC(N(C)C(c3cnc[nH]3)=O)C(C)(C)C2)=O)ccc2nnnn2c1 N1(C(C2C(C)CC2)=O)CC2CN(C(=O)C3CCc4scnc43)CC(C1)O2 c1(CC(CCC)O)nc(-c2ccccc2C(F)F)nn1C1CCS(=O)(=O)C1 N1(C(C23CC(C(=O)NC)(C2)C3)=O)CCN(C(CCC(=O)O)=O)CC1 CC(C)C(C)(C)C(=O)NC(C1CCCN(C(c2ccc(F)o2)=O)C1)C C(N=c1nc(C2CC2)[nH]s1)C1CN(C(=O)C=Cc2cnc[nH]2)C1 Cc1cc2[nH]c(C(=O)NC3CN(C(=O)CCOc4cccnc4)CC3C)cc2s1 CCS(=O)(=O)c1ccc(C(N2CCCC2CN(C(=O)C2=CCCS2)C)=O)cc1C C(C(F)(F)CCNC(=O)COC(F)F)n1cc(Cn2c(C)ccn2)nn1 C1(C(=O)NCCCN(C)C(c2ccccc2[N+](=O)[O-])=O)CC2(C1)C(F)(F)C21CC1 c1(C(=O)NC(C)CN(C(=O)CN2C(=O)CCCC2=O)C)ccc2ccncc2n1 c1(NC)cc(C(N2CCCN(C(C3(CC4CCC4)CC3)=O)CC2)=O)cc(Cl)n1 N1(C(c2c(N)ccc(C)c2)=O)CC2CCC(NC(C3CC(C(C)C)C3)=O)CC2C1 C1(CNC(C(C)C(F)(F)F)=O)CN(C(c2cc(Cl)no2)=O)CCC1(F)F C12(C(=O)NC3CCC(CNC(C=CCOCCOC)=O)CC3)CCCC(C)(C1)OC2 C(=O)(CC(C)(C(F)F)N(C)C)NCCc1nc(C(C)NC(C2CCCC2)=O)sc1 Cc1cc(C(=O)NC(C)C(C)(C)NC(C2CN(S(C)(=O)=O)C2)=O)ccc1C(C)C c1(C(=O)NC2C(NC(C=CCC)=O)CS(=O)(=O)C2)cnc2c(c1)nc(O)n2C N1(C(CC(C=C)(C)O)=O)CC2(COC(CNC(=O)COc3ccc(Cl)cn3)C2)C1 N1(C(C2CCC(CNC(c3scc(C)n3)=O)C2)=O)CC2CCN(C)CC2C1 c1(C(C(=O)NCC)N2CCC2C2CCCC2)ccnc(Cl)c1OC C(=O)(C(C)(C)C(=O)NCC1CCN1C(C1(C2CC2)CCC1)=O)NC C=CC(C)CCN=c1[nH]c(=NCc2cn(CC)nn2)c2sccc2[nH]1 C1(C(N2CC=CC(C(=O)NCC(=O)OC(C)C)C2)=O)C2CCC(C2)C1C C#Cc1ccc(C(=O)NCC(C(=O)NC2CC2CN(C)C)N(C)C)cc1 N1(C(C(CC)C)=O)CC(NC(=O)C(COC)N(CC)Cc2ccccc2)CC(F)C1 CN1C(=O)CN=C1NC(c1csc(-c2cccnc2)n1)=O c1(COC)ccc(CNC2CCC(C(=O)NCc3cccc(F)c3)CC2)c(Cl)n1 C1(CCOC)(NC(=O)CC2CCCO2)CCN(C(C2CCCO2)=O)CC1 CC(C)(C)C(C#N)C(=O)NC1CC(C(F)C(=O)NC2CCC(O)C(O)C2)C1 CC1CC(CCC(=O)N(C)CCF)CCN1C(=O)CN1CCN(C)CC1 N1(C(c2ncc(CC)nc2)=O)CC(CNC(c2coc(Cl)c2)=O)OC2CCCC12 C1(C)(C(=O)NCCC(CNC(c2c(CC)cccc2)=O)O)CC(C(C)C)=NO1 c1(C(=O)NC(C(CO)NC(c2cnc(C(=O)OC)s2)=O)C)cccn2cnnc12 c1(C(N2CC(NC(c3ccc(C)nc3O)=O)C(C)C2)=O)cc2c(C)cccc2o1 C1(C)(C(=O)NC(C)C(O)C(F)F)CCN(C(c2cc(Cl)c[nH]2)=O)CC1 C1(NC(C2C(C=C)C2)=O)CCC12CCN(C(C13C4C5C1C1C3C4C51C)=O)CC2 C(=O)(CCCCN=[N+]=[N-])NC(C(C)C)CNC(C1CC1(F)F)=O C(c1ccc(Cl)c(C(F)(F)F)c1)=CC(N1CC2C(N)CC(C2)C1)=O c1(OC(C)C(=O)NC2C(C(=O)NCc3ncccc3F)CCC2)cccc(F)c1 C#CCCCCCCC(=O)N1CCN(C(=O)C(C)Cc2cccnc2)CC(O)C1 C1(CC(=O)OCC)CCCN1C(=O)CCc1ccc(C(=O)OC)[nH]1 CC1(C)C(C(N2CC(CNC(c3ccoc3Cl)=O)C(C(F)(F)F)C2)=O)C1(C)C c1(CC)nccnc1C(=O)NCC(C)(CNC(=O)Cn1ccnn1)OC c1(NCC(N2CC=CCC2c2cccnc2)=O)cc(OC(F)(F)F)ccc1O N1(C(c2c(C)cncc2)=O)CC(C)(C)CC1CNC(c1cnc(C(F)(F)F)s1)=O C1(NC(C(=C)C(F)(F)F)=O)CN(C(=O)CN2CCNC2=N)C2(CCOC2)C1 N1(C(C(=O)NCCc2ccccc2)=O)CCC2C(CCC(=O)N2C2CC2)C1 C1(C(=O)NC(c2ccccc2)c2ncon2)(OC)CCN(C(C(=O)O)C2CC2)CC1 c1(C(F)(F)F)nc(C(F)(F)F)[nH]c(=NC2C=CCCC2)n1 CC1CN(C(=O)CCNC(=O)CO)CC1CNC(c1cccc(C2(C)CCC2)c1)=O C=CCC(CNC(=O)C=CCC1(NC(C2CC=CC2)=O)CCC1)CC(C)C C1(NC(C(CC2CCC2)NC(c2cc[n+]([O-])cc2)=O)=O)CCCC(O)C1O C1(CNC(=O)Nc2cc(N3CCN(C)CC3)ncc2)CNc2ccnn2C1 C(=O)(C(C(C)C)NC(=O)CCn1cccc1)N(C)CC N1(C(c2c(C)con2)=O)CCC(C)(C)C(C(=O)NC(CCO)C(C)C)C1 N1(C(C(CCC)(C)O)=O)CCN(C(=O)C(CC)(CC)CO)CC12CC2 N1(C(CC=C)=O)CCC(C(N2CC(CO)C(C)(C)C2)=O)C12CCC2 CC1(C)CN(C(c2cnc(O)o2)=O)CCC1C(=O)NCC1CC1(C)C c1(CC(=O)N(CC(CN(C(=O)C=Cc2cscn2)C)O)C)csc(S)n1 N1(C(C2CC=C(C)CC2)=O)C2CC1CN(C(=O)Cc1nc(C)no1)C2 S(=O)(=O)(c1c[nH]ccc1=NCC1C(C)(C)C1(F)F)N(C)Cc1c(C)ccc(C)c1 N1(CCNC(CC2CCN(C(COC3(C)CCC3)=O)C2)=O)CCNC(=O)C1 C(=O)(C(F)C(C)(C)O)N1CCC(CC=C)(NC(=O)CCc2ccc(NC)cc2)C1 C(C(N=[N+]=[N-])C(=O)N1CCCC1CC(=O)NCCC(Cl)Cl)OCC N1(C(C(C=C)OC)=O)CCC(NC(=O)C(C2CCC2)OC)CC(C)(C)C1 c1(NCc2c(=N)[nH]cnc2)[nH]c(=NCC2CC(O)C2n2cccn2)nc2sccc12 N1(C(C2ON=C(C)C2)=O)CCN(C(=O)Cc2ccc(F)cc2C)C2COCC12 Cc1nccc(OC(C)(C)C)n1.N12CCN(CC1)CC1CC1N(CCC(=O)O)C2=O c1(C(N2CCN(C(C3C(Cl)(C(=O)OC)C3)=O)CC2C)=O)cc2ccccn2c1 C12(C(=O)NCC3N(C)CCN(C(c4ncnn4C)=O)C3)CC(C)(C1)OC21CCC1 N(C(=NCCCF)NCC1CCCN1C1CC1)CCC(=O)N(CC)CC C1(NC(c2ccc(C(F)(F)F)s2)c2nnnn2C2COC2)CCC2(CC2)C1 C(=O)(C1=CCCSC1)NCC(CCOC)NC(C(CC)n1cncn1)=O N1(C(CCC2N(C(C3CC(OC)(OC)C3)=O)CCC2)=O)CCOC(C)(C2CC2)C1 c1(CC)cccnc1C(=O)N(C(C)(C)CC(=O)N(C1CC(O)C1)C)C N1(C(C=CCOC)=O)CCC2(CCC2NC(C23CCC(=O)N2CCS3)=O)CC1 C(C(CC(=O)NC1C2CCCOC12)NC(=O)CCc1cn(C)cn1)OC C1(NC(c2ccc(C)cc2)=O)(CNc2ccccn2)CC2CCC1CC2 CC(C)(C(=O)NCC(CO)NC(=O)CNC(c1cccs1)=O)c1ccncc1 c1(OC)nccnc1C(N1CCC(CNC(C2CC(=O)CO2)=O)C1)=O C1(C(N2CCN(C(C#C)C)CC2)=O)CCN(C(=O)C(C)C)C12CCC2 N1(C(c2nccc(C)n2)=O)CCCC(NC(c2cc(C)oc2C)=O)CC1 c1(-n2cc(COCC(=O)O)nn2)cc(F)cc(F)c1 c1(OC)ccc(C(=O)N(CC(O)CNC(=O)CC(C)n2ccnc2)C)cc1F Cc1ccc(C(=O)NC2CCCC(C(C)NC(=O)C3CC3)C2)nc1 N1(C(CN2CCN(C(c3c(C)cnn3C)=O)CC2)=O)CCC(CO)CC1(C)C CC1(C)CCN(C(c2cc(CCO)on2)=O)CC1CNC(=O)CC1CCOC1 C1(O)(CC(C)C)CCN(C(=O)C(C)N(C(c2coc(C(F)F)c2)=O)C2CC2)C1 n1(CC)cc(C(N2CCC2(C)CC(=O)NCC2(C)CC2(F)F)=O)c(C)n1 c1(CNC(C(C2CCCC2)OCC)=O)ncccc1CNC(=O)CCCOC c1(NC(CN(C(C2(CC#C)CC=CCC2)=O)C)C)c(F)cc(C#N)cc1[N+](=O)[O-] C1(C)(C(=O)NCC(=C)C)CN(C(c2cnc(O)n2CC)=O)C(C)(C)C1 C1(CCNC(c2cc(-c3ccccn3)no2)=O)CCN(C(=O)Cc2cn[nH]c2)C1 C1(CC(=O)NCCCCN(C(C2(CC=C)CCC2)=O)C)CS(=O)(=O)C1 C(=O)(C(C)CCCC(C)=O)N(CCN(C(CCCCCC#C)=O)C(C)C)C C1(CC(=O)NC(CC=C)CNC(c2cn(C3CC3)nn2)=O)CCC2(CCC2)O1 C(=O)(CCCCC(=O)NC(CCC1CCC1)C(=O)NCC1C=CCOC1)OC c1(OC)cccc(C(N2CCC(C(=O)N(CCCO)C)(CF)C2)=O)c1C c1(C(N2CC(C)C(NC(C3CC(=O)N(C)C3)=O)C2)=O)ccc(F)c2ncccc12 Cn1cc(C(=O)N(CCCC(=O)O)CC2CC2)c(O)n1 C#CCC(O)C(=O)N1CC(NC(c2cc(C)n(CC(F)(F)F)n2)=O)C(SC)C1 C=CC(C)(CCOC)C(=O)NCCCN(C)C(C1CCc2nccn2C1)=O C1(C(=O)NCC(=C)CCNC(c2ccc(=NC)[nH]c2)=O)CC2CCC(C1)C2(F)F CCC(C)C(O)C(=O)NCC1CCN(C(c2ccc(CO)cc2OC)=O)CC1 C(=O)(C(F)(F)C(F)(F)F)NCC1CC(CNC(=O)CC(=O)NCC2CC2)OC1 c1(C(N2CCOCC(NC(C(CCC)C)=O)C2)=O)ccc2c(c1F)CCC2 CC(C)(C)CC(C)(C)C(=O)NC1CC2CC1N(C(C1CCCO1)=O)C2 N1(C(CC(=O)NCC#C)=O)CCOC(C(NCP(C)(=O)OCC)=O)CC1 c1(OC)cc(F)c(-c2cn(C(C)CNC(=O)CCCC(=O)C3CC3)nn2)c(F)c1 c1(C(N2C(C)(C(=O)NCC3CCCC4CC34)CC(O)C2)=O)cc2ccncc2[nH]1 C=CCCCCC(=O)NC1CC(CCNC(C2COCCC2(F)F)=O)C1 c1(NC(c2c(-c3c(OCCC)nccc3)cncc2F)=O)cc(Br)c(C)cc1O c1(CC(N2CCC(CCC(=O)N(C(C)C)CC)C2)=O)cc(C)n(C)n1 C1(NC(CNC(C)=O)=O)CC2CCC1CN(C(c1ccc(NC(C)=O)cn1)=O)C2 CCS(=O)(=O)CCCCCOC1CCN(C(=O)OC(C)(C)C)C(C)C1 N1(CC(=O)N(C(C)CNC(=O)CCc2cnc(O)[nH]2)C)CCP(C)(=O)CC1 C(=O)(CC(F)(F)C(F)(F)F)N1CC(NC(CCCCC#N)=O)C2(C1)CC2 N#Cc1cc(N(C(c2ccc(Cl)c(O)c2)=O)CC2CNC2)ncn1 C1(CNC(C(C)CCO)=O)CCC(C)N(C(=O)CC2CCC(F)(F)CC2)C1 c1(Nc2ccnc(SC)n2)ncnc2[nH]cc(I)c12 Cc1ccc(C(=O)N(C2CCN(C(=O)C(C)Cc3ccccc3)C2)C)c(O)c1C C1(N(C(=O)COC2(C)CCC2)CCC)CCN(C(c2cnccn2)=O)CC1 c1(C(N(CCCN)CCO)=O)ccc([N+](=O)[O-])s1.C(CC=O)=CC=C CC1(C(N2CCCOC(CNC(=O)CCC3CC3)C2)=O)CCCNC1=O C(=O)(C(C)(C)C(C)(C)C)N1CCC(CNC(c2c(CC)occ2)=O)(OC)CC1 C1(NC(C(CC)N(C)C)=O)CCN(C(C2CCSCC2)=O)CC(C)(C)C1 CCC(CC(=O)NC1(CO)CN(C(c2ccc(C(C)=O)o2)=O)C1)C1CC1 N1(C(CSC)=O)CCC(CCC2CCCN(C(C34COCC3C4)=O)C2)CC1 c1(C(=O)NCC(C)NC(c2cnc(C3CC3)[nH]2)=O)cnn(-c2ccncc2)c1 C=CC(C)(O)CC(=O)N1CC(NC(=O)CSc2nnc(S)s2)CCC1C CC12COCC1(C)CN(C(C1C3CN(C(=O)CC(F)(F)F)CC13)=O)C2 c1(Nc2ncncc2I)cccc(S(=O)(=O)N2CCCC(O)(C(C)C)C2)c1 C12(C(=O)NC3CCC(NC(C(C)(C)c4cccs4)=O)C3)CC3CC1C2C3O C1(C(=O)NCCN(C(c2c(C(=O)OCC)n(C)nc2)=O)C)CC2(CCC2OC)C1 c1(C(N(CCNC(=O)Cn2cnnn2)CC)=O)cc2c(O)ccc(F)c2[nH]1 C(=O)(C1=CS(=O)(=O)CCC1)NC(CCCC)CNC(=O)CCc1cnco1 C1(NC(=O)NCc2c(C)ccc(N3CCNC3=O)c2)Cc2ccccc2C1O CCC1CCN(C(=O)C(C2CCCCC2)F)c2cc(Br)ccc21 N1(C(CSCC)=O)CCC(N=c2[nH]c3ccccc3cc2[N+](=O)[O-])CC1C C1(NC(CN(C)C2CC2)=O)CC2(CCC(CNC(c3cn(C)nn3)=O)CC2)C1 N1(C(C(Cc2cc[nH]n2)NC(CC(CC)O)=O)=O)CC2(CCC2)CC1C c1(C(=O)NCCCOCCN(C(C(=O)N(C)C)=O)C)oc2ccccc2c1CO c1(NC(NNC(c2cc(C)c(Br)cc2)=O)=O)nc2c(s1)COCC2 C(=O)(C(O)CN(C)C(C)=O)N(CC(C)NC(=O)CCSC)CC Cc1ccc2occ(C(N3CC(NC(c4cnncc4C)=O)CC(O)C3)=O)c2c1 c1(C(N2CC(NC(C3CCCN3)=O)C2)=O)scnc1-c1cnn(C2CCOC2)c1 c1(OC)cc(C(C(=O)NCc2ccc(Cl)cc2)N(C)CC2CC2C)ccc1SC N1(C(C2(C(C)C)COC2)=O)CCC(C(C)NC(=O)CNC(=O)CNC(N)=O)CC1 c1(C(=O)NC(C2CCN(C(c3c(C)ccc(F)c3)=O)C2)C)n[nH]c2c1COCC2 C1(CNC(c2cccc(CC)n2)=O)CN(C(c2ccc(NC)cn2)=O)CCC1C C1(C(N2CC(O)(CNC(C34CCC(CC3(F)F)C4)=O)C2)=O)CC2(CCCC2)CO1 CC1=C(C(=O)NCC2CC23CCN(C(=O)C(C)(C)F)CC3)C(C)(C)CCC1 C1(NC(C2CCN(C(CC)=O)C2)=O)CC12CCN(C(c1cc(C#N)[nH]c1C)=O)CC2 CC(C)(C)C(CNC(c1cc(C2CCOCC2)on1)=O)NC(C1(O)CCOC1)=O C1(N(C(C(CC)=CC)=O)CC)CCCN(C(=O)CC2CC(C)(C)CCO2)CC1 C1(C(N(CCCOCCNC(COCCCC#C)=O)C)=O)CNC(=O)N1 C1(CNC(c2cnc(OCC)nc2)=O)C2CCCC1N(C(=O)C(C)CCOC)C2 C1(C)(CC)C=C(C(=O)NC(C2CCN(C(=O)Cc3cc(O)nc(O)n3)C2)(C)C)C1 Cc1nc(N2CC(C(C)NC(c3cnnc(O)c3)=O)C2)cc2nncn12 CC(CCNC(=O)CSC(F)(F)F)NC(=O)CN(C)C(=O)OC(C)(C)C c1(C(N(CCNC(CCN(C)CC)=O)C(C)C)=O)cncc2n[nH]cc12 C1(C)(C(=O)NCC(C)CN(C(=O)CSCc2cccs2)C)C=CCCC1 CCC(C(=O)N(CCCNC(c1cscc1F)=O)C(C)C)OC1CCCCC1 C(=O)(CC(C)(CN(C)C)C(F)(F)F)NC1CC(C)N(C(=O)CC2=CCCC2)CC1 CCCCCCC(C)(C)C(=O)NC1CCC(C)N(C(=O)CCc2cc(C)on2)C1 c1(C(N2C(C)(CC(=O)Nc3ccn(CCOC)n3)CC2)=O)ccc(C2CC2)cn1 N1(C(c2ccc(CC)s2)=O)CCN(C(=O)C2=C(Cl)CCC2)C2CCCCC2C1 C#Cc1ccc(C(=O)NCC2CC(CNC(c3nnc(C)s3)=O)CO2)cn1 c1(C(N2CC=CC(NC(C3N(C(C)=O)CCC3)=O)C2)=O)cc(O)nc(O)c1 C(=O)(C1=CCCCCC1)NC1CN(C(C=Cc2n(CC)ncc2)=O)CC1F C1(CNC(=O)Cc2cnsc2)CCCCC1C(N1CCC1CC1CCCC1)=O C(=O)(CCC(C)S(C)(=O)=O)N1CCC(C2CC2)(CNC(c2c(C)ncs2)=O)C1 c1(CC2(C(N3CCC(NC(C4CC=CCO4)=O)C3)=O)CC2)cccc(Cl)c1 Cc1cnc(C)c(C(N2CCCC(Cn3cc(-c4cnsc4)nn3)C2)=O)c1 C1(CNC(c2cnc(O)o2)=O)CN(C(c2cccc(C3CCC3)c2)=O)CCCO1 c1(C(N2CCC(NC(=O)Cc3c[nH]nc3O)C(F)C2)=O)ccc(F)c2ccoc12 c1(CC(=O)NC(C2CCCCC2)C(C)NC(c2cocn2)=O)ncccc1F C(C(CC(C)C)C(=O)NC(C)(CC(C)C)C(N)=O)NC(C(CO)OC)=O C1(CN(C(CC2C(C)C2)=O)C)CCN(C(C2CC(=O)CCO2)=O)CC1 Cc1nsc(C)c1C(N1CC(C(N2CCOC(C(N)=O)C2)=O)C1)=O c1(C(C(=O)N(C(C)CNC(c2csc([N+](=O)[O-])c2)=O)CC)C)ccc(F)cc1F c1(CCC)ccc(N)c(C(=O)NCC(CC)NC(=O)C(C)Sc2nncn2C)c1 c1(C2(C(N3CC(C(C)NC(C4CC(C(F)F)C4)=O)C3)=O)CC2)ncccc1F N1(C(C(F)OC)=O)CCCCC(NC(c2ccncc2O)=O)C1 N1(C(c2cccc(SC)c2)=O)CCC2(CNC(=O)C#CC(C)C)CCCCC12 N1(C(C2N(C(C)=O)CC(O)C2)=O)CC2CCC(C1)N2C(c1cncc(C)c1Cl)=O CCCC(C)CC(=O)N1CCCC(C)(NC(=O)CC2=CCCC2)C1 C(=O)(C1CC(=O)N(C)c2ccccc21)N(C1CCC(CNC(CC)=O)CC1)C C1(OC)CCCC(C(N2CC3CC2C3CNC(c2nn(C)cc2Cl)=O)=O)C1 C(C(C)C(=O)NC1CCC1CNC(c1ccns1)=O)OCC C1(NC(c2ccc(F)c(F)c2)=O)CCSC12CN(C(c1ccc(F)cn1)=O)C2 C1(N(C)C(c2ccnn2C)=O)CCN(C(C2CCCN2c2ncccn2)=O)CC1 C1(CN2CCC(NC(COCCCC)=O)C2)CCC2(CCC2)O1 c1(NC(C2C3CC2N(C(c2cccnc2Cl)=O)C3)=O)ccc(I)c(F)c1 CC1C(NC(=O)C(C)(C)c2ccno2)CCCN1C(=O)CCCC1CCC1 N(C1CCc2c(Cl)cc(Cl)cc21)C(N1C(c2ccc(OC)cc2)CC(C)C1)=O c1(CC(=O)NC2(CNC(C34CC(CO3)C4)=O)CCC2)cccc(O)c1 N1(C(CC2C(C)(C)C2)=O)CCC(O)(CNC(C2CCCC(O)C2)=O)C1 N1(C(CC2N(C)CCOC2)=O)CC2CC(C1)N(C(c1cccc3nn[nH]c13)=O)C2 c1(CCNC(c2ccc(-c3ccc(NCCO)cc3)cn2)=O)cc(F)cc(F)c1 C=CC(C)CC(=O)NCc1ccsc1C(N1CCOCC1COC)=O C(C(=O)Nc1cncc(CO)c1)(C(C)(C)C)NC(c1nccc(CC)c1)=O N1(C(CN(C)C)=O)CCc2onc(C(N3CCC4NC(=O)OC4C3)=O)c2C1 C(=O)(CC(CN(C)C)CC)N1C(CN(C(C2(CC#C)CC2(F)F)=O)C)CCC1 C1(C(N(C2CCN(C(c3cccnc3O)=O)CC2)CCC)=O)CC(F)(F)C1(C)C N1(C(CCC(C)C)=O)CCC(C2(O)CN(C(=O)CSC(F)F)C2)CC1 c1(CC)cccc(C(=O)N(CCNC(N2CCCC(CC3CC3)C2)=O)CC)c1F c1(OC)cccc(S(=O)(=O)CCNC23CCC(CC2n2cc(C)cn2)C3)c1 N1(C(c2cc(Cl)cs2)=O)CC2CC1CN2Cc1cnc(C(F)F)s1 C1(NC(c2cn(C)nn2)=O)CN(C(c2sncc2Br)=O)CC1F c1(Nc2c(-c3ccn(CCOC)n3)cnc(OC)c2)cc(C)c(Br)cc1[N+](=O)[O-] CN1CC(CCNC(=O)COC2(C)CN(C(=O)C(O)C3CCCC3)C2)CC1=O c1(C(=O)NC2C(n3cc(CCC4N(C)CCC4)nn3)CCC2)cccnc1Cl C#CC1CN(C(=O)C2=CCC(NC(=O)CCCn3cccn3)C2)CCO1 C(CCF)(C(=O)NC1CC(OC)C1)NC(c1cc(COC)[nH]n1)=O C(C(C)(C)CNC(c1nn[nH]c1Cl)=O)N(C(=O)C(=O)NCC1CC1)C N1(C(COCCCC#C)=O)CCCC2(NC(c3oncc3CC)=O)CCCC12 c1(C(=O)NCC2(OC)CN(C(=O)CCC(=O)N(C)C)C2)cc(F)cnc1O C1(NC(C(C#C)(C)C)=O)CCCN(C(c2ncccc2OC)=O)C1C C1(CC=C)(C(=O)N(C2COC(C)C2)C)CCN(C(=O)COc2ccsn2)C1 Cc1ccc(-c2nc(CNC3(C)CC(C(=O)O)C3)cs2)cc1 c1(NC(CC)Cc2ccc(C)cc2)nccc(=NCCc2c[nH]nc2C(F)F)[nH]1 N1(C(C(CCC)(C)O)=O)CC2CCC1CN2C(C12CCCC1C2(F)F)=O C(=O)(CCC(N)=O)NCCOCC(=O)NC(C(=O)OCC)C c1(CC(=O)NCCN(C(c2cnc(C)s2)=O)C)sc(O)nc1O CCC(C)C(CC(=O)NC1CC(C)(C)C1)NC(C1(C)CC=CC1)=O C=CC(C)CC(=O)N1CCC(C(N2CCC(N3CCCC3)C2)=O)C1 c1(C(N(C2C(NC(CCSCC)=O)CCCC2)C)=O)cc(Cl)c2[nH]c(O)nc2c1 N1(C(C2(COC)CN(C(C(CC=CC)C)=O)C2)=O)CC(O)CC(O)C1 C1(C(N2C(C(=O)OC)COCC2)=O)CN(Cc2cccc(SC)c2Cl)CCC1O c1(C2C(NC(c3cn(C4C(OCC)COC4)nn3)=O)CCO2)ccc(Cl)c(F)c1 c1(C(C)C)ccc(C#N)c(N(C2CN(C(=O)CC3(C)CC3)C2)C)n1 C1(OC)(CNC(C2CCCC2(C)C)=O)CCN(C(=O)CCNC(=O)NC)C1 C(C(F)(F)C(C)(C)O)NC(C(CCC)NC(=O)CCc1ccnn1C)=O c1(N2C(C)(CNC(c3ccc(CC)s3)=O)CCC2)ncnc2cc(C)[nH]c12 C1(C(=O)NCC2CCCN(C(C=CC=CCC)=O)C2)CCCS(=O)(=O)N1 c1(COc2cccc(C(=O)OC3C=CCCC3)c2)c(F)cccc1Cl Cc1cccc(C(=O)NCCCC(C)NC(=O)CCOCC2CCCO2)c1N C1(C(C)NC(=O)CC2CC(F)(F)C2)CCN(C(=O)CSCC2CCCCO2)CC1 N1(C(CN(C)C2CC2)=O)CCC(C2(NC(c3ccc(=O)oc3)=O)CC2)C1 c1(CC=C)cccc(Br)c1C(=O)OCCNC(=O)C(C)C CN=c1cc(C(N2CCN(C)CC2CNC(=O)CC(C)(C)OC)=O)cc[nH]1 Cc1c(Cl)ccc(C(=O)NCCC2CCCCN2C(C2CCOC2C)=O)c1N C1(CN(C(=O)C(O)COCc2ccccc2)C)CCCCN1C(=O)CC1CC1 c1(C(N2CC(O)(CNC(C3CC3c3ccccc3)=O)C2)=O)cc(O)cc(Cl)c1 Cc1cc(C)c(-c2ncc(CN3CCN(C4CCCC4O)CC3)s2)c(C)c1 C(=O)(CCC(=O)N1CC(NC(c2ccc(-c3ccccc3F)[nH]2)=O)C(C)C1)OC C1(OC)(CNC(c2cc(F)n[nH]2)=O)CN(C(C2CC=CCC2)=O)C1 C1(NC(C(c2ccc(Cl)cc2)C)=O)CC2CCC1N(C(c1cnnc(Cl)c1)=O)C2 CCCC(C(=O)NCCNC(=O)OC(C)C(C)C)NC(C1CCCSC1)=O Cc1ccnc(C(N2CCC(N3CCN(C(c4cc(C)[nH]c4C)=O)CC3)C2)=O)n1 CC1=NNC(=O)C1CC(N1CC(CNC(=O)CNC(=O)NCC2CC2)C(C)C1)=O N1(C(C2(CN(C)C)CCCC2)=O)CCCC(C2CN(C(c3ccc(F)o3)=O)C2)C1 C1(C(=O)NC(CC#C)CCOC)CC(C)(C)CCN1C(c1ccc(C)cn1)=O C1(NC(=O)CC(F)F)COC2(CCN(C(c3cncc(O)c3Cl)=O)C2)C1 N1(C(C2(COC)CC2)=O)CC2CCCC(NC(c3ccc(C)nc3OC)=O)C2C1 N1(C(c2nc(C(C)NC(CC(C=C)C)=O)oc2)=O)CCCC(OC)CC1 CCS(=O)(=O)C1CCN(C(c2cccnn2)C(=O)NCc2cccc(Br)c2)C1 c1(C(N2CC(NC(COCC(C)(C)C)=O)(CO)C2)=O)ccc(Br)c(N)n1 C(CCCC(=O)NC1C(C)CCC1C)N(C(Cc1ccn(CC)n1)=O)C C1(CNC(=O)CC2CCCOC2)CN(C(c2cnsc2)=O)CCC12CCOCC2 C12(C(N(CCCC)CCCO)=O)CC1CCN2C(c1scnc1CC)=O C(=O)(C(CC(F)F)NC(=O)Cn1cccc1)NCC(C)(C)CCO c1(CCC(=O)NC2C(OC)CN(C(C(CC(C)C)O)=O)C2)cnc2n1CCCC2 c1(OC)cccc(C#N)c1NC(C12CC1CN(Cc1cscn1)C2)=O C1(NC(CC(n2c(CC)ncc2)C)=O)CCCC2CN(C(C3CCOC3)=O)CC12 n1(CC(=O)NC2C(CNC(CNC(=O)OCC)=O)CCC2)cc(P(C)(C)=O)cn1 CCCCCCC(=O)N1CCCC1C1C(NC(=O)CSCC(N)=O)C1 Cc1cc(C(F)(F)F)nn1CC(=O)N(C(C)CN(C)C(C1CC2CCC2C1)=O)C CC1=C(C(=O)N2CCN(C(c3cn(CC(N)=O)nn3)=O)CC2CF)CCS1(=O)=O c1(C(=O)NC2(CNC(=O)Cc3cocn3)CC2)ccc2cccnc2c1F N1(C(C2COCCN(C(C(C)(C)OC)=O)C2)=O)CC2CCC(CO)(C2)C1 c1(NCCCC2C(C)C2)ccc(S(=O)(=O)NCC2(C)OCCO2)c2ccncc12 C(=O)(CS(=O)(=O)Cc1cccs1)N(C1CCN(C(C=NOC)=O)CC1)C N1(CCC(C(=O)OCC)C(=O)OCC)CC2CCC(C1)C21OCCO1 N1(C(C2CCCC(N(C)C)C2)=O)CCCCC(NC(C23CC(F)(C2)C3)=O)C1 c1(CN2C(C(=O)NCc3c(C)cccc3)CCC2)ccc([N+](=O)[O-])cn1 C1(CC=C)(C(=O)N(CCN=[N+]=[N-])CC)CCN(C(=O)CC2CCCC23CC3)C1 C1(C(N2C(C)(CNC(C3C(C)CCC3)=O)CCC2)=O)C2CCC1(C)C2(C)C C(=O)(C1=CCCCCC1)N1CCN(C)C(CNC(c2ccnn2C(C)(C)C)=O)C1 N1(C(C(C)SC(C)C)=O)CCOCC(NC(c2cncnc2C2CC2)=O)C1 N1(c2cc(C(C)C)ncn2)CCN(C(=O)Cc2cc(Br)ccc2O)C2(CC2)C1 C1(CCNC(C(C)CC2CC2)=O)CCCN(C(=O)COc2cccc(Br)c2)C1 N1(C(CCn2ccc(C)n2)=O)CCC2(CCN(C(=O)C(C)c3ccn[nH]3)C2)C1 C1(C)(CNC(c2c(C)nc[nH]2)=O)CCCN(C(=O)C(c2cc(Cl)cc(Cl)c2)=O)C1 C1(C)(C(=O)NCc2n(CC)ncn2)CN(C(=O)C(C)S(C)(=O)=O)C(C)(C)C1 C1(NC(CC2(C=C)CC2)=O)CCCC12CCN(C(C1CC(N(C)C)C1)=O)CC2 C(C(C)(C)CC(=O)NCC1(C#N)CC1)NC(C1(C(C)(F)F)CC1)=O CCC(C)(C(=O)NC1CCCC1NC(=O)COc1cccc(C)c1)OC c1(CC(=O)NC2CCC(O)(CCCC)CC2)c(C)oc2ccccc12 c1(N(C2(O)CCSC2)C)ncc(C(C)(C)O)cn1.N12CCC(C1)C2=O c1(CN2C(C(=O)Nc3ncn(C)n3)CC(OC)C2)cc(Cl)cnc1F N1(S(c2ccc(NCC3CCC(C)(C)O3)nc2)(=O)=O)CCc2ccc(F)cc2C1 c1(C(=O)NCCCCC(C)NC(c2cncc(C)c2)=O)c(N)c(F)cc(F)c1F C1(NC(C2(SC)CN(C(C3CCCSC3C)=O)C2)=O)CCC(O)CC1 C1(C)(C(=O)NCC(C)NC(CC=C(C)C)=O)CCCCC1(F)F C(c1cnn(C)c1C)=CC(N1C(CCCC)CCC1)=O.C1(C2CN2)CN1 C1(C(=O)NCC2C(CNC(c3cc(C(CC)C)no3)=O)C2)CCCCC(=O)N1 c1(C(=O)OCC)ccc(Cl)c(O)c1S(=O)(=O)Oc1ccc(C2CCC2)c(Cl)c1 c1(CC)[nH]nc(C(N2CCC(O)(C(C)NC(c3cc(OC)no3)=O)C2)=O)c1C C1(CNC(C=C(C)C(C)C)=O)CC(O)CN1C(C1CC2CCC1O2)=O C(=O)(C(C(C)(C)C)N(C)C)NCC1N(C(C(c2cnn(C)c2)C)=O)CCOC1 C1(CNC(CCc2c(C)n[nH]c2C)=O)CCN(C(=O)CC(C)F)C12CC2 c1(OC)ncnc(C)c1C(=O)NCC12CC(NC(c3occc3C)=O)(C1)C2 C1(CC)CC(C(=O)NC(C2CN(C(c3csc(C4CC4)n3)=O)CCO2)C)CCO1 C(=O)(C#Cc1cccc(Cl)c1)OC(c1c(F)cccc1F)C c1(CC)nn(C)c(CNC2C3CCC(O3)C2C(N)=O)c1Cl CC#CCCCCNC(C12CC1CN(C(c1sccc1F)=O)C2)=O C1(c2n(C)ncc2)CN(C(=O)NCC2CCCS(=O)(=O)C2)CC(=O)N1 C1(C)(NC(CN(C(C(n2ccc(C)n2)C)=O)CC(C)C)=O)CCC2(CC1)CC2 C(C(C)(CC(=O)NCC1(c2cccc(Br)c2)CCOCC1)C(F)(F)F)N(C)C c1(C(=O)OC)ccc(O)nc1N1CCCC(NC(=O)C(C)OC)C1 N1(C(C(c2cn(C)nn2)NC(C(CC)=CC)=O)=O)CC(N(C)C)C2(CC2)C1 c1(Cc2cn(C(C)CNC(c3ccc(CCF)cc3)=O)nn2)cc(C#N)c[nH]1 C=CC(C)C(C)C(=O)NCC1(CCNC(c2csc(N3CCCCC3)n2)=O)CC1 C1(CNC(c2n(CC(=C)C)nnn2)(C)C2COC2)CCC(F)(F)C(C)(C)O1 Cc1c(O)ccc(C(=O)NC2CCC(NC(=O)Cc3cccs3)CC2)c1C CC(CC(=O)NC1CC(CCC(N)=O)C1)C(C)(C)NC(=O)CCCC1CCC1 CC(CC(=O)NC(CO)C(N1CC2CCC2C1)=O)CC(C)(C)C CCCCCCC(=O)N(C)CC1(O)CCCN(C(=O)CC2CC2(C)C)C1 c1(CC(N2CC3C(CNC(C4(C(F)F)CC(=C)C4)=O)(C3)C2)=O)cccc(C#N)c1 C1(CNC(C(COCC)C)=O)CCCC(NC(c2cn(C)nc2C(C)C)=O)C1 C(C(C)C)(C(O)C(=O)N1CC(C)(C(=O)NC2(C)CCC(C)CC2)C1)OC C1(C(=O)NC(CC)CC2CCCC2)CCc2c(nnn2CC)C1 C1(NC(C(CC)C)=O)CC2CCC(C1)N2C(C1C=CCN(C(=O)OC(C)(C)C)C1)=O Cc1c(F)ccc(C(N2CCN(C(c3cc[nH]n3)=O)C3CC23)=O)c1C#N CC1CCN(C(c2cccc(CO)c2)=O)CC1CC(=O)NOC(C)(C)C C(=O)(C(CC)C(F)(F)F)NCC(CC)NC(c1ccc(C#N)cc1F)=O N1(C(=O)Nc2csc(C(F)(F)F)n2)C2CCCC1CC(N1CC3CC3C1)C2 N1(C(C2C(C(N)=O)C2)=O)CCCC(C2CN(C(c3ccc(F)c(Cl)c3N)=O)C2)C1 c1(SC)c(C(=O)NCC2COCCN(C(C3CC4(CC4)C3)=O)C2)cccc1F Cc1c(CNC2N(C(=O)Nc3ccccc3)CCNC2=O)cccc1O CN1CCN(C(c2cn3ccnc3s2)=O)C(CNC(C2C=CCC2)=O)C1 c1(CC(=O)NCC2CC(N(C)C(C3CCCOC3)=O)C2)ccc(O)cc1 C1(C(N2CC(C(N(CC)CC)=O)C2)=O)CC(O)CN1C(=O)CCC1CC1(Cl)Cl CCC(C)(C)CC(=O)N(C)CC1CC1.c12ocnc1CN1CC2C1 C12(NC(c3c(C)c[nH]c3)=O)CCC(C(N3CCC(F)(CO)C3)=O)(CC1)C2 C1(N(C)C)(CO)CC(C)CC(C)(C)C1.C1(C)CN=C(NC2CCC2)NC1CC Cn1nnc2cc(C(=O)NC3CCCC(CNC(c4ccco4)=O)C3)ccc12 c1(C(N(C(C)CCNC(c2ccc(CF)cc2)=O)C)=O)[nH]nc2ncccc12 C1(NC(CSC)=O)CC(NC(=O)CNC(=O)NCC(N2CCCC2)=O)C12CCC2 C1(CC(=O)N(CC(COC)O)CC2CCC2)CCOCC1 C(C)(C)(CC(=O)NOC1CCN(C)CC1)N(C(C1=CC(C)(CC)C1)=O)C c1(C(N2CCC(CC(=O)NCCCn3c(C)ncc3)C2)=O)cc(Br)cnc1F N1(C(c2ccnc(C(C)C)n2)=O)CCC2(CC1)CC2NC(=O)CC(F)F N1(C(CC(C)C)=O)CC(CCNC(=O)C(C)(C)NC(c2ccccc2)=O)OC(C)C1 c1(C(N(C2CN(C(=O)CC(O)c3ccccc3)C2)C)=O)ccc(N)c(F)c1F Cc1cc(F)c(C(=O)NCCCOCCNC(=O)CCc2ccnn2C)c(Cl)c1 c1(C(=O)NC23CC(NC(CCS(C)=O)=O)(C2)C3)ccc(F)cc1Br c1(NCc2c(C)nc3ccccn32)ncc(S(=O)(=O)N2CCSC2)cc1Cl c1(COC(c2n(C)ncc2)=O)ccc2c(=O)[nH]ccc2c1 C(=O)(C(F)C(C)(C)O)N(CCNC(C(C(=O)OC(C)(C)C)OC)=O)CC1CC1 c1(C(=O)NCC2N(C(COCCCOC)=O)CC2)sccc1OC(F)F c1(CSCC(=O)OCCc2ccc(Br)cc2)cnc2ccccc2c1 CN1CCN(CC2CC3(CC(NC(=O)NC4CC(C5CCC5)C4)C3)C2)CC1=O c1(CC)noc(C)c1C(=O)NCCn1cc(CNC(=O)C=Cc2cnn(C)c2)nn1 c1ccccc1Cl.C(C(C)(C)NC(C1CCC1C(N)=O)=O)NC(COCC)=O C(CNC(=O)Cc1csc(C(=O)OC)n1)(CC(C)C)NC(c1nc(CC)oc1)=O c1(C(N2CC(CC(=O)OC)OC(C)C2)=O)cc(F)c(N)cc1Cl c1(C(=O)NCC(C2CC2)NC(C(C)(C)CC#N)=O)c(Cl)ccc(Cl)c1Cl C=C(Br)CC(C)(C)C(=O)NC1CC1NC(C1CC1C#N)=O C1(CC(=O)NC2(c3ccccc3)CN(C(C=C(C)C)=O)C2)CCCN(C)C1 C1(C(=O)NC(CC=CC)CO)CC2(CC2)CN1C(=O)C(=O)C(C)(C)C c1(CNC(C2C(NC(CC3(C)CCOC3)=O)COC2)=O)ccc(Cl)cn1 C(c1ccc(C)cc1)=CC(=O)NC(C(=O)NCC1(OC)CCOC1)c1ccco1 C12(C(N(CCCNC(CN(CC(=O)OCC)C)=O)CC3CC3)=O)CCC(OC)C1C2 N1(C(c2ccc(C)o2)=O)CC2CC(NC(c3sccc3Br)=O)CC2C1 C12(CNC(C(=O)NCC(F)(F)F)=O)CCCC1CCN2C(C1CCC=CCC1)=O c1(C(=O)NCCN(C(CN(c2nccn2C)C)=O)CCOCCO)ncn(C)n1 c1(OC)c(CC(N2CC(NC(=O)Cc3cncn3C)CC(C)C2)=O)cccc1Cl c1(OCC(C)C)cccc(C(=O)NC(C2(O)CN(C(C3CC=CC3)=O)C2)C)c1 C(=O)(CCC(C)NC(=O)C(C)N1CCCC1)NCC1(CC(C)C)CC1 Cc1ncc(C(N2CC(N(C(=O)CC3CCC(=O)N3C)C)C(C)(C)C2)=O)c(C)n1 c1(C(N(C(CCNC(C2C(C)CC=CC2)=O)C)C)=O)cc2scc(Cl)c2[nH]1 Cc1nn(C)c2nc(C(N3CC(NC(=O)C(F)C(C)C)CC(C)C3)=O)ccc12 c1(C(CNCc2nnnn2CCC2CC2)OC)ccc(N(C)C)cc1.C1(N)CSC1 c1(CC)nc2sc(C)cn2c1C(N1CCC(NC(=O)C(C(C)C)N(C)C)CC1)=O C12(NC(C(CCCC)=O)=O)CCCC1CN(C(c1c(C(F)(F)F)n[nH]c1C)=O)C2 C1(CNC(C(CC2CCC2)NC(C)=O)=O)CN(C(C2CC=CC(O)C2)=O)CC1(C)C N1(C(C(C)=C(CC)C)=O)CC=CC1(C(=O)NCCn1ccccc1=O)COC CC1CCN(C(=O)C=CC2CCCN2C)C(C(=O)NCc2ncc[nH]c2=O)C1 c1(C(=O)NCC(=O)NC(CCCC)CNC(=O)CS(N)(=O)=O)cc2c(s1)CCCC2 C(C(C)(C)C(=O)OCC1CCCC(N(C)C(C2CC(C#N)C2)=O)C1)OC CC1(CNCc2sc(N3CCCCC3)nc2Cl)CSCCO1 N1(C(C(CC)C(F)(F)F)=O)CCCC2(C1)CN(C(c1nc(C)n(C)n1)=O)CCO2 C(=O)(CCC(=O)NC(C)CCNC(=O)CCn1cc(C)cn1)NCCC N1(C(COCC)=O)CCC(C2CC2)C1CNC(c1c(F)ccc(F)c1F)=O C1(NC(Cc2ccc(CCCCC)cc2)=O)CN(C(=O)C(C)(F)F)CCC1CO C1(C)(CC)C=C(C(=O)NC2CC(CO)N(C(C3CC(=C4CCC4)C3)=O)C2)C1 CC1C(NC(C2CN(S(N)(=O)=O)C2)=O)CCCN1C(C1C(F)(F)C12CC2)=O N1(C(Cc2cc(C)nn2C)=O)CCOCC(F)(CNC(=O)C=C2CCCCC2)C1 Cc1nn(C)c2c(N3CC(C)SC(C)C3)nc(=NCC3(C)CCOCC3)[nH]c12 c1(SC)cc(C(=O)NCC2CCC(NC(=O)CCC3(C)CC3)C2)c(C)o1 c1(OC(C(CC=CC)NC(=O)OC(C)(C)C)=O)cc(C(C)=O)ccc1F c1(CNC(=O)Nc2c(C)cns2)cc(-c2cccc(Cl)c2)n(C)n1 c1(NCc2cc(C)n(C)n2)[nH]c(=NCCCOc2nccs2)nc2ncn(C)c12 C(=O)(CS(=O)(=O)CCC)N1CCC=C(CNC(c2nc(CCC)oc2)=O)C1 c1(NC(C2(O)CCC(C)CC2)=O)cc(Br)cc(I)c1F c1(C(C)=O)c[nH]c(C(=O)NC(C)(C)CNC(C2CC2c2cnnn2C)=O)c1C C(=O)(CCCC(=O)NCC1(O)CCN(C(C2CCCC(C(N)=O)C2)=O)CC1)OC C(C(F)(F)C(=O)NC(c1ccc(F)cc1)CNC(=O)CC1CCC(C)CC1)OC N1(C(CC2(C(=O)NC3CC3)CC2)=O)CCCC(C(=O)NCCCN(C)CC)CC1 Cc1nn2ccccc2c1C(=O)NCCCCN(C(=O)CCC(C)C=O)C C1(C(C)C)OCCCC1C(=O)NCCC1CSCCN1C(c1ccc(=N)[nH]c1)=O c1(C(N(C2CCN(C(c3cc(F)n(C)n3)=O)C2)CCC)=O)ccc(C(F)F)cc1 N1(C(c2cncc(OC)c2)C(=O)NC2(C)CC2)CCCOC(C)C1 CC1(C)CC(CNC(C2CC2c2cccc(O)c2)=O)CCC1 C(=O)(C1=CC(C)(CC)C1)N1C(CC=C)(C(=O)N(C)CC2(CO)CCC2)CCC1 Cc1sc(O)nc1C(=O)NC1CN(C(=O)C(F)=CCCF)CC1n1cccn1 C1(C(=O)NC(C(C)NC(c2cnnc(O)c2)=O)CO)CC2CCC(C1)C2O C=C(Cl)C(C)(C)C(=O)N1CC(CCNC(C2(C(F)F)CCC2)=O)C(C)C1 N1(C(COCCCC)=O)CCC2(CC1)C(NC(=O)C(C)C(F)F)CS2(=O)=O c1(C(=O)NC(CCCC)CNC(=O)C(F)(F)c2cscn2)cnc(O)n(C)c1=O Cc1c(NCCCc2nccc(O)n2)nc[nH]c1=NCC1CC1CO C(=O)(CC(CCCC)NC(c1cc(O)cc(F)c1)=O)NC1(CC=C)CCOCC1 c1(N2CC3C(C)C3C2)nc2ccsc2c(=NC(C)COCC(F)(F)F)[nH]1 c1(C(=O)NCC2(C(=O)OCC)CCC2)ccccc1-n1cncn1 C(=O)(C1c2c[nH]nc2CN1C(C1OC2CCC1C2)=O)NCc1cc(C(C)C)n[nH]1 C1(F)(C(=O)OC)CN(C(=O)NC(C2CC2(C)C)C)CC1C1CC1 CC1(O)CCNCC1.C12CCC(C1)NC2=O.c1(C2(C=O)CC2)cnccn1 C1(NC(=NCCCCl)NC2CCCC2)CCC2(CCCCC2)C1 N1(C(c2cnc(SC)s2)=O)CCC(C)C(NC(=O)C(C)Oc2cccc(C)c2)C1 N1(C(Cn2c(C)ccn2)=O)CCCC(C2CCCN2C(c2cc[nH]n2)=O)C1 CCCCC(C)C(=O)N1CCC(NC(=O)Cc2csc(=N)[nH]2)CC1 C1(NC(=O)C(O)C2CC2)CC2CC(NC(C3CC(F)(F)C3)=O)C1C2 N1(C(C(=O)NCC2C(CNC(C3CC(OC)C3)=O)C2)CC)CCc2ccccc21 C(=O)(CCS(C)=O)NCCC(Cc1ccccc1)NC(CCc1scc(C)n1)=O C=CC1CN(C(c2csc(=N)[nH]2)=O)CC1NC(c1cc(CO)n(C)n1)=O CC(C)CS(=O)(=O)CCC(=O)N(CC(O)CNC(=O)CC1(O)COC(C)(C)C1)C c1(C(=O)NCC2CCN(C(CCC3C(C)(C)C3)=O)C2)cc2ccccc2o1 C(=O)(C(F)(CNC(C1CC(CF)C1)=O)C(C)C)NCC1(C)ON=C(C)C1 Cn1c(C(=O)N2CCC(C(=O)NC3CCC(C)(C)C3)O2)ccc1C#N c1(N(CCOC)CCNC(=O)CCc2ccccn2)ncnc(Cl)c1[N+](=O)[O-] N1(C(C2N(C)CCCC2)=O)CC2CN(C(c3ncc(Br)cc3O)=O)CC2C1 CC(CCCNC(C1CC1(C)C)=O)NC(=O)C(F)Cc1ccccc1 c1(C(N2CCN(C(CC3CC(=C)C3)=O)C(C)C2)=O)c(C)nn2c1CCCC2C c1(C(=O)NC2CC3CN(Cc4ccc(Cl)nc4)CC3C2)cc2cccc(Cl)c2[nH]1 CC(C)C(C(=O)NC(c1nncn1C)C)NC(C1CC(C)(C)C1)=O C12(C(=O)NCC3(OC)CCCC3)C(NC(=O)CCc3ccnn3C)C3CC1C2C3 c1(CNC(C(C)OCC)=O)cc(C(=O)NOCCCF)co1 CC1(C(=O)NC2CCCCC2NC(=O)CCc2ncc[nH]2)CCNC(=O)C1 c1(C(=O)NCC(CNC(COCCOC)=O)C)c(O)nnc(CO)c1CC c1(CC)[nH]nc(Cl)c1C(N1CCN(C(C)CNC(=O)C(C)N2CCCC2)CC1)=O c1(C(=O)NCC(CNC(C2CC(C)(O)C2)=O)F)ccc(-c2coc(O)n2)cc1 c1(C(=O)NC(CCNC(C(c2ccnn2C)C)=O)C)cc2n(c1)CCS(=O)(=O)C2 C(CC(C)C(=O)N(CCC(C(C)C)NC(=O)CSc1ccccc1Cl)C)=CC N(C(=NCCc1cc(O)cc(Br)c1)N1CCC(F)(C#N)C1)C(CC)CC C(=O)(C1=CCCOC1)NCc1c(C(N(C2CCN(C(=O)C3CC3)C2)C)=O)cccc1 C1(NC(c2ccc(CC)c(C)c2)=O)CC12CCN(C(=O)CCCF)CC2 N1(C(c2cc(CCC)on2)=O)CCC(C)(C)C1CC(=O)NC(C)CC(C)(C)OC Cc1cc(CO)oc1C(=O)NCCC1CCN(C(C2CC(n3cccn3)C2)=O)C1 C12(C(N(C3CC3)CC3N(C(CC4(CSC)CC4)=O)CCC3)=O)CCC(F)C1CC2 c1(C(=O)NCC2CN(C(C3CCC4(CC4)C3)=O)CCCO2)cccc2[nH]ncc12 N1(C(CC)COC(C2CC(C(C)C)C2)=O)CCN(Cc2ccc(OC)cc2)CC1 N1(C(C#CC(=O)N(C)C)=O)CCC(NC(C2CC(=O)N(C)C2)=O)CC(O)C1 CCC1=NOC(C(=O)NC2COCC2C(=O)NC(C)C(C)C)C1 n1(C(C(=O)OC)C)nnnc1C(c1conc1C1CCC1)Nc1cccnc1 N1(C(C(C=C)c2ccccc2)=O)CCOC2(C1)CN(C(C1CC1C1CC1)=O)C2 Cc1sc(C(=O)NCC2CC(NC(C3(C)CC3C)=O)C2)cc1S(N)(=O)=O C1(C(F)(F)F)(C(=O)NCC(C)NC(C(CC)OCC)=O)CC2CC2C1 C(=O)(C1=C(C2CCCOC2)N(C)C(=O)NC1c1cc(OC)ccn1)OCC CCS(=O)(=O)CC(=O)N(CC(O)CN(C(=O)C(c1cccc(C)c1)(F)F)C)C c1(C(=O)NCC(C)N(C(CCOCCOC)=O)C)coc2c(Cl)cccc12 Cc1cc(=NC(=O)CC2CC(F)CN2C(C2CC(=O)N(C)C2)=O)[nH]n1CCO C1(C)(COC)CCCN1C(C1(CCN(C)C)CC1)=O.C12CC(C1)NC2=O C1(NC(c2c(C)nsc2)=O)CN(C(=O)C(C)Sc2ccccc2)CC1C#N C1(CCCNC(C(C)OCCC(C)C)=O)CCCN1C(=O)CCc1cncs1 CC1CCCc2nc(C(=O)NC3(C4CCCN(C(c5cc[nH]n5)=O)C4)CC3)cn21 c1(C(=O)NC(C)CNC(c2ccc(CC(C)C)s2)=O)cccc(C2CCOC2)c1 Cc1nc(NCCSC2=NOC(C)(C)C2)cc(=NC(C)C2CN(C)CCO2)[nH]1 c1(C(=O)NC2CC(F)(CC)C2)cc(NC(C2CCC(C)(CC)O2)=O)cc(F)c1 Cc1cccc(N)c1C(=O)NC1(C)CN(C(C2CC(OC(C)(C)C)C2)=O)C1 c1(OCC)ccc(C(=O)NC23CC2CN(C(=O)C(C)NC(C)=O)C3)cc1C#N C1(C(=O)NCC(C2CCCCC2)NC(C2CC(CC)(CC)C2)=O)CC(C)(C)CO1 c1(COC)nc(C)ncc1C(N1CCN(C(=O)C2=CCOC2)C2CC12)=O C1(O)(CC(=O)NC2CC(C)N(C(C34CC(C3)C4)=O)C2)CCN(C)CC1 c1(C(N2C(C(C)C)C(NC(=O)C(C)C(C)(C)C)CC2)=O)cnc2n1CCCC2 N#Cc1ccc(Br)c(NC(C2CC23CN(C(c2nc4ncccn4n2)=O)C3)=O)c1 C1(NC(C(C)n2cccn2)=O)CCN(Cc2cncc(Br)c2)CC1(C)C C(=O)(C(CCC(C)C)N(C)C)NC1C(NC(COCCCC)=O)C1 C(N=c1[nH]c(=NCCN2C(=O)CCC2=O)[nH]c2cc[nH]c12)C1CCC(=O)NC1 c1(C(N2C(C)(CCC)CC2)=O)coc2c1CN(C(=O)C(c1ccn(C)c1)C)C2 c1(CNC(C2OCCN(C(C=C(COC)C)=O)C2)=O)cc(C)cc(C)c1 C(=O)(C(C)S(=O)(=O)C(C)C)N1C(CNC(c2cccc(CC)c2)=O)CN(C)CC1 Cc1ccc(C(=O)NCC(N2CCC2CNC(=O)C(F)=CC2CC2)=O)cc1 C#CC(C)(C)C(=O)NC(CCN(C)C(C1CC2(CCC2)C1)=O)C(C)C C1(C(=O)NCCN2CCC3CC23)CCCN(C(=O)CC2CC2C2CC2)C1 CCC(CC)C(C)C(=O)NC1CN(C(c2c(C(F)(F)F)cnn2C)=O)C1 Cc1cc(C(F)(F)F)cc(C)c1NC(C)CC1CCOCC1 C(=O)(C#CC1CCCCO1)N(CC(O)CN(C)C(c1ncc[nH]c1=O)=O)C N1(C(C(C)OCCCC)=O)CC2C(CN(C(=O)CCc3cn(C)cn3)C)C2C1 N1(C(Cc2cn(CC)nc2)=O)CCCC(C)(C(=O)NCC2CN(C)CCO2)C1 CCCCC(CCC)N=c1[nH]c(=NC(C)c2ncn(C)n2)c2c(F)cccc2[nH]1 C(=O)(C(C)C(O)C(C)C)N1CCCC(CNC(c2c(C)cc(SC)o2)=O)C1 Cc1cc(Br)ccc1CN1CCCC(C)(C(=O)N(C)CCc2cccc(Cl)c2)C1 C1(CNC(CN(C(=O)C(C)OCC2CC2)CC)=O)(CO)CC2CC2C1 C=CCCCC(C(=O)N(C)CC1(OCC)CCC1)NC(C1CCOCC1)=O CCCCCC(=O)NCc1cccc(CN(C(=O)Cc2nn(C)cc2Cl)C)c1 C1(C(=O)NCC2(C(N)=O)CN(C(CC3C(C)CCCC3)=O)C2)CCC(N=[N+]=[N-])C1 C1(CNC(C2CCCC2C(N2CCCC(CCF)C2)=O)=O)CC(C2CC2)=NO1 C1(CN(C(=O)CCNC(N)=O)CCCN(C(=O)CCC2CCC2)C)CCCCC1 C1(c2n(C)ccn2)CN(C(=O)COC2CC2)CCN1C(=O)COc1nccs1 C1(C)(CC)C=C(C(=O)NCC2CC(O)CN2C(c2cc(C(C)(C)C)n[nH]2)=O)C1 CC1CCC(C)(C)CN1C(C1CCCN(C(=O)CSC(F)(F)F)CC1)=O N1(C(C(C)=CC)=O)CC2CC2(CNC(C2CCCN2C(=O)NC)=O)C1 C1(NC(C(C2CN(C(c3ccn(COC)n3)=O)C2)O)=O)CNC(=O)C1(C)C C(=O)(C1Cc2ccccc21)N(CCCCCCNC(C1N(CC)CCOC1)=O)C c1(C(=O)NCC(C)(CO)NC(c2c(CC)cc[nH]2)=O)oc(C)cc1C c1(C(N(CC(CN(C(C(c2cccc(Cl)c2)C)=O)C)O)C)=O)cccnc1O C(=O)(C(C)CC(=O)c1ccc(F)cc1)N(C1(CO)CC2C=CC1C2)C c1(C(=O)NC(C(C)NC(c2cc(CF)on2)=O)C)c(O)cnc2ccc(Cl)cc12 N1(C(C2(CC=C)CCCC2)=O)CCC(NC(c2ccn(CC)c2C)=O)C(O)C1 c1(C(C(=O)NCCCF)N(CCC#N)CCC)cccc(COC)n1 c1(CCNC(C2C(COC)C2)=O)ocnc1CNC(C1CC1C)=O C(c1cc[nH]c1)=CC(=O)N(C(C(=O)NCCC#CC)C)C c1(N2C3CN(C(C4C(C)OC(C)C4)=O)CC2CC3)nc2c(cc1C#N)CCC2 N1(C(C(COC)OC)=O)CC2CCCC(NC(=O)C(C)N3CCC3)C2C1 C(=O)(CC(C)C(F)(F)F)NCC1C(NC(C2N(C(C)=O)CCC2)=O)CCCC1 N1(C(c2n(COC)ncc2)=O)C2CCC1C(C)C(NC(c1n[nH]cc1C)=O)C2 c1(Sc2c(C(=O)NC3CC(OC)C3(C)C)cccc2)c(F)cccc1F C1(NC(C=Cc2n(CC)ncc2)=O)CCN(C(C23CCCCC2C3)=O)C(C)C1 N1(C(CCC2CC(NC(c3c(OC)c[nH]n3)=O)C2)=O)CCN(C(C)=O)CC1 C1(NC(Cc2nc(C)sc2C)=O)CN(C(C2(C)CCCCC2)=O)CCC1C c1(OC)ccc(Cl)c(NC(C2CCN(C(=O)C(c3ccccc3)=O)CC2O)=O)n1 Cc1c(C(=O)NCC2CCC(NC(c3cnn[nH]3)=O)CC2)[nH]c2cc(Cl)ccc12 C1(N(C(=O)CC2CC=CC2)C)CCCN(C(c2ccc(C(C)(F)F)cc2)=O)C1 N1(Cc2n(C)cnc2-c2ccccc2)CCC2(CC1)CC2C(=O)O N1(C(C(CC)SC)=O)CCCCC1CCN(C(=O)CCCOC(C)(C)C)C c1(NCc2c(OC)ccs2)cc(C(F)(F)F)c(Br)cc1[N+](=O)[O-] N1(C(CCCC#C)=O)CCC(CO)C(NC(c2cc(C)nc(C(F)(F)F)n2)=O)C1 C1(C(=O)NCCc2scc(C)n2)C2CC3C(C2NC(C2CC(=O)NC2(C)C)=O)C13 c1(C(=O)OCC(C(C)(C)C)=O)nc(C(F)(F)F)n2ccccc12 N1(C(COC)=O)CCC(O)(C(C)CNC(C2(SC)CCC2)=O)C1 C(=O)(C(C)(C)CC(C)C)N1CCC(n2cc(C(c3ccccc3)OC)nn2)C1 N1(C2C(NC(CCOCC#C)=O)CCC2)CCN(C(c2nocc2CC)=O)CC1 c1(C(C)C)cnc(Cl)nc1N(C)CCO.c1(COC(F)F)ccccc1 c1(CC(=O)NCC(CC=C)NC(C2CC2CF)=O)cccc(Br)c1Cl C1(CNC(c2ccc(NC)cc2)=O)CC2CCC1N2C(=O)CC(C)C(F)F c1(C(N(CCCNC(=O)C(C)SC)CCC)=O)cccc(CC)c1 C1(C(=O)NC(CC=C)C)CCCN1NC(=O)CN1CC(=O)NC1=O C1(NC(c2c(CC)csc2)=O)CC2(C1)CC2NC(c1cnn(CC)c1CC)=O C1(C(=O)NC2CC3CC(NC(C4CCC=CCC4)=O)C2C3)CC2(CCOCC2)C1 N1(C(c2c(C)nc[nH]2)=O)CCC(C)N(C(C2CCC(F)(F)CC2)=O)CC1 c1(C(=O)NC(C2CN(C(=O)CCN(C)CCO)C2)C)nccnc1-n1ccnc1 c1(CC(CNC(=NC)NCC(F)F)CO)c(F)cccc1F CC1CC(NC(=O)CCC2CC2)CN(C(=O)CC2CSC2)C1 CCC(F)(F)C(C)(C)NC(=O)C(C1(O)CN(C(C2COC(=O)N2)=O)C1)F C(C(C(=O)NC(c1ccc(Br)cc1)C#N)C(F)(F)F)SC S(=O)(=O)(c1cccc(NC2CCN(CC(F)F)C2)c1)NC1C(=O)CC1 C(=O)(CCN=C(NCCc1ncn(C)n1)NCCn1ccc(C2CC2)n1)NC N1(C(c2cnc(CC)s2)=O)CCC2(CCCN(C(c3[nH]ccc3C)=O)C2)C1 N1(C(C(C)(C)F)=O)CCN(CC(=O)NCc2cccnc2Br)CC1 n1(C(C)C)nccc1-c1cn(C2CCC(C(=O)NCC34CC(F)(C3)C4)C2)nn1 c1(C(N2C(C(N3CC(C)C3)=O)C3CC(F)C2C3)=O)ccc2ccc(Cl)cc2n1 C1(CC(=O)NCCC2CC(NC(CCSCC)=O)C2)CCOC(C(C)C)C1 c1(C(N(CC(C)NC(C2(CO)CCCCO2)=O)C)=O)ccc(F)cc1[N+](=O)[O-] Cc1cccc(Cl)c1C(=O)NC1(CNC(=O)CC2CC3CCC2CC3)CCC1 ClC=CCN=c1nc2sccc2c(NCC2CSCCS2)[nH]1 C(=O)(NNc1ccc(C#N)cc1C(F)(F)F)NC1C(C(C)C)CCC1 c1(C(=O)NCCN(C(C(CC=C)CC)=O)C(C)C)nnn2c1CSCC2 C(=O)(CC(CC#N)c1ccccc1)N1CCC(N(C(C2CCOC2)=O)CC)CC1 c1(C(N2CCC(=CCNC(C(C(C)O)C)=O)CC2)=O)cnc2c(c1)COC2 C1(CNC(C=CSC)=O)CN(C(=O)Cc2cc(C3CC3)on2)CCC1C(F)(F)F c1(OC)ccc(C(C)C(=O)NCC2CCN2C(=O)C=Cc2ccoc2)cc1OC C1(NC(C2CCCN(C(C(C)OCC)=O)CC2)=O)C2CCOC2C1(C)C Cc1c(C(N2CCC(O)C2C(C)(C)C)=O)[nH]c2cc(Cl)cc(Cl)c12 Cc1cc(CC(=O)NC(CNC(C23CCCC(CO2)C3)=O)C2CCC2)cc(F)c1 C(=O)(CCCCC1CC1)NC1C=CC(C(=O)NCC(C)(C)O)C1 C1(NC(Cc2c(C)noc2Cl)=O)CCN(C(C2(C)COC2)=O)CC1(C)C c1(C(C)(C)C)cc(C(=O)NCCC2CC2C2CC2)n(-c2ccc(F)cc2)n1 C1(C2CCOCC2)(C(=O)NC(CC)CNC(=O)Cc2ccsc2Cl)CC1(F)F c1(SCC)cccnc1C(=O)NCC1C=CCN1C(=O)Cc1ccsc1Br c1(C(C)O)ccc(NC(=O)CC2CSCCS2)cc1 N1(C(C23N(C(=O)CCc4cnoc4)CCC2C3)=O)CCC2(CCOC2=O)C1 C1(NC(C2N(C(c3nc(CC)oc3)=O)CC2)=O)(CO)CCC(C)(C)C1 c1(CCC(=O)NCC=CCNC(C2C(CC)C2)=O)c(F)cccc1F C(=O)(CC(C)(C)NC(=O)C(O)C(C)C)N(CC#C)CC1CC1 C1(C(=O)NCc2ccc(CNC(c3nc(C)n(C)c3)=O)cc2)CNC(=O)CC1C C1(C)(C(=O)NC)CCN(C(=O)C(Cc2ccoc2)NC(=O)Cc2ccn(C)c2)C1 CC1CCC(CC(=O)NCc2ccoc2C(=O)NC2(CC3CC3)CCC2)O1 CC1CCN(C(C23CCCCC2C3)=O)CC1NC(c1ccn(CCF)n1)=O c1(CC)ccc(O)c(C(N2CC(CNC(=O)CCCOCC)C(C)C2)=O)c1 c1(C(N2CC(F)CC(NC(C(C)CC(N)=O)=O)C2)=O)n[nH]c2c1CCCCC2 c1(OCC(=O)NCC)ccc(C)cc1OC.C12CN(CC1C)C(=O)CC(=O)N2 Cc1cc(=NC2CN(C(=O)C(C)CC(C)C)CC2C)nc(-c2cccs2)[nH]1 n1(CC2(C)CC2)nc(CCO)nc1-c1cnc(-c2ccco2)s1 C1(CC(=O)N(C23CCCC2C3)C(=O)CN2CCCCCCC2)CC2CC(=O)C1C2 C1(NC(C2(C)CC2F)=O)CC2(CCC(NC(c3cc[nH]c(=N)c3)=O)CC2)C1 c1(CCC(=O)NC(c2ccccc2O)C)cccc(OC2CC2)c1 C1(c2ccccc2)(NC(C=CS(C)=O)=O)CCN(C(=O)CC(F)(F)C(F)(F)F)C1 c1(C(N2C(CNC(C(CC)(C)CC)=O)CCC2)=O)ccc2nc(O)nc(O)c2c1 C1(C#N)(NC(COc2c(OC)cccc2)=O)CCN(C(c2cnccn2)=O)C1 c1(CNC(=O)CC2CN3CCC2CC3)n[nH]c2c1CN(C(c1ccsc1)=O)CC2 n1(CC(=O)N(CCOC)CC)ccnc1C.C1(=O)CN1.C1(C)CNC(=O)N1 C1(NC(c2c(C)n(C)cn2)=O)CCN(C(c2ccoc2CC(N)=O)=O)CC1O c1(N2CCC(C(=O)NC3C4C(=O)C5C(C4)C53)CC2)ccc([N+](=O)[O-])cc1 C1(O)(C(C)NC(CSCC#C)=O)CCN(C(c2cc(C(F)F)ccn2)=O)C1 N1(C(=O)Cc2ccc(OC(F)F)cc2)CC2CCN(C(=O)C(O)C3CC3)CCC2C1 c1(OC)cc(C)cnc1C(=O)NCC(C1CCC1)NC(C1(C(C)(C)O)CCC1)=O c1(CNC(=O)NC(c2n(C)nc(CC)c2Br)C)ccc(F)c(Cl)c1C N1(C(c2c[nH]c(=NC)s2)=O)CCC2(CC2C(=O)NCc2cc(C3CC3)on2)C1 CC1OC(=O)NC1C(=O)N(CC(O)CNC(=O)CCN1CCC(O)CC1)C N1(C(CN(CCC#C)C)=O)CC(NC(c2c(Br)ncn2C)=O)CCC1C O(NC(=O)CCC1CCOC1)C(C(=O)OCCC(C(=O)OC(C)(C)C)(C)C)(C)C CC(CC(F)(F)F)C(=O)NCC(C)N(C)C(c1cc2cccnc2[nH]1)=O c1(C(=O)NC23C(n4cc(C(CCC)=O)nn4)CC(CC2)C3)cccn2nncc12 c1(N2CCC(NC(c3ncc(OCC)nc3)=O)CC2C)ncc([N+](=O)[O-])cc1Br C(=O)(C(C)(C)CO)N(CC(CC)NC(C1CC(OC(C)C)C1)=O)C CCC(CC)C(=O)NCC(N1CC(CF)(NC(=O)CCc2cc(C)[nH]n2)C1)=O c1(C(N2CCCC(NC(C(C)CSc3ccccc3)=O)C2)=O)ccn2ccsc12 N1(C(c2ccc(C(=O)OC)nc2)=O)CCC2(CCN(C(C34COCC3C4)=O)C2)C1 C1(N)(CCCC(=O)NC(c2ncc(C)s2)CC)CCOCC1 C#CCC(C(=O)NC)C1CC1.c1(C(N2CC(CC=C)(OC)C2)=O)ccccn1 c1(C(=O)NC2CN(C(CSC(C)C)=O)C2)cc(C(F)(F)F)ccn1 CC(C)CCCCCC(=O)NC(CC(=O)NC(CO)CCCO)C(C)(C)C c1(C(N2CC(C)CC(NC(CC(C)(C)OC)=O)C2)=O)c(C)[nH]cc([N+](=O)[O-])c1=O C(=O)(CC(CC1CC1)NC(C1CCC1)=O)NCC=CCOCC CCC(CCOC)C(=O)N1CCOC(CNC(c2ccc(C(O)CF)cc2)=O)C1 CC(C)C(C(=O)NC1(CO)CN(C(=O)C(C#N)C2CC2)C1)c1ccc(Cl)cc1 C12(CNC(c3c(C)occ3)=O)CCCC1CCN2C(=O)Cc1ccccc1 CCCC(C)CC(=O)N1CCCC(NC(c2cn(C)nc2COC)=O)C1 c1(OC)ncc(C(N2CCC3CCC23CNC(c2cccnn2)=O)=O)cc1Cl c1(NCCN2CCC(OC)C2)nc[nH]c(=NCC2CN(C)CCO2)c1C c1(CC=C)cccc(C(=O)NC(C)CC(C)NC(=O)CCC(C)OC)c1 N1(C(C(C2CCOC2)OCC)=O)CCN(C(=O)Cn2cc[n+](C)c2)CCC1C C(=O)(C1=CCCC(C)(C)C1)N(CC(CC)NC(=O)CCC1CCCOC1)CC C#CC1CN(C(C23CC(CN(C(=O)C(CCC)OC)C2)C3)=O)CCN1C C1(NC(C(CC(C)C)O)=O)CN(C(C2CCCN2S(C)(=O)=O)=O)CC12CCC2 c1(C(CC)(C)C)ccc(C(=O)NCCNC(c2cc(C)oc2C(F)(F)F)=O)cc1 CC(C)S(=O)(=O)C(C)C(=O)NCC1CC1CNC(c1ccncc1F)=O c1(OC)cc(C)c(CN2CCC(C(=O)NCc3cncc(Br)c3)C2)cc1C c1(C(N(CCCNC(CC(COC)C)=O)C(C)C)=O)ccc(Cl)c(F)c1 C1(C(=O)OC)CCC(C(=O)N(C)CCN(C(=O)C(F)n2cccn2)C(C)C)C1 c1(OC)ccc(CC(N2CC3CC2(CNC(=O)C2=CCCC2)C3)=O)c(F)c1 N1(C(C2C(CCOC)C2)=O)CCN(C2CN(C(=O)C(C)OC)C2)CC1 O=c1ccc2cc(CN3CCOC(c4ccc(F)cc4F)C3)ccc2o1 N1(C(c2cc(C(C)=O)on2)=O)CCC(O)(CNC(C2CCCCC(=O)N2)=O)CC1 C(C)(C)(CC(F)C(=O)NC(c1ncc(C)cn1)C)NC(c1cc(CC)no1)=O C1(NC(C2CCS(=O)(=O)N2)=O)CN(C(C2(CF)CC2(F)F)=O)CC2(CCC2)C1 N1(C(C(CCC)C)=O)CCC(C2CCCN(C(=O)C(c3c(C)noc3C)C)C2)C1 c1(C(=O)NCC2(O)CCCN(C(CS(C)(=O)=O)=O)C2)nccc2c[nH]nc12 C1(CNC(c2c(CC)ncnc2)=O)COCCN(C(c2ccc([N+](=O)[O-])o2)=O)C1 CC(CC(=O)N(C1(CC(=O)NCCCn2cccn2)CC1)C)C(F)F Cc1nn(C)cc1C(=O)NCc1ccc(CN(C)C(C2CCCNC2=O)=O)cc1 c1(CNC(C(C(C)O)C)=O)nn(C)c2c1CN(C(C1CC(=O)N1)=O)CC2 c1(C2C(C(=O)NCC34C(CN(C(CCC)=O)C3)C4)C2)ccc2ccccc2c1 C(=O)(C#CC1CCCCO1)NCC(C)(CC(C)C)NC(CCC(=C)Cl)=O CCCCCCCCCCC(c1nnnn1C(C)(C)CC)NC1COCC1CO N1(C(c2ccn(-c3ccc(Br)cc3)n2)=O)CCOCC1C(N1CCCC1)=O C12(NC(C3COCC3c3ccccc3)=O)CC1CN(C(=O)CC1CC(F)(F)C1)C2 c1(CN2CC(CC(=O)Nc3c(OC)nc(C)nc3)C2)ccc2ccc(O)cc2c1 CC1(C)CCC(C)(C)N(C(c2cc3cc(Cl)ncc3s2)C(=O)NCCCF)C1 c1(C(N(CCNC(=O)C2=CCCS2)C2CC2)=O)nn(-c2ccccc2)ccc1=O C=CC1(C(=O)NCc2cc(C)cnc2F)CCN(C(C2C3CC(=O)CC23)=O)CC1 Cc1cccc(NC(C)C(N2CCOCC2CNC(c2ncccc2Cl)=O)=O)c1 Cc1cc2c(=O)n(Cc3c(C)cc(Br)cc3Cl)cnc2cc1F C1(NC(C2(Cc3ccon3)CC2)=O)CC2CCC(C1F)N2C(=O)C(O)C1CC1 C1(NC(C(CSC)OC)=O)CN(C(=O)CN(c2ccnc(Cl)n2)C)CC1O C1(C(=O)NC23CC(CNC(C4C(=C)C4C=O)=O)(C2)C3)OCCC1(C)C.OCC C1(CC(=O)NCCCc2cc(C)no2)CCCC(NC(=O)CC(C)(F)F)C1 C(CC(C)C)(C(=O)N(C)CC1CN(C(=O)CC2CCC(=O)NC2=O)C1)NC(C)=O C(=O)(CC(C)N1CCCC1=O)NCC(CC)N(C(CCOCC)=O)C C1(C(=O)NCC)CC2(CCN(C(c3cccc(-c4ccsc4)c3)=O)CC2)C1 c1(C(=O)NC2CCCC(CNC(Cc3nnc(C)o3)=O)C2)cc2n(c1)CCCC2 C(C(C(C)C(C)C)NC(c1ccc(N)c(Cl)c1)=O)NC(c1c(C)scc1)=O Cc1onc(C(=O)NC2CCCCC2NC(c2cc3cscc3s2)=O)c1[N+](=O)[O-] CCC(CC)C(C(=O)NC1(CNC(=O)CC(C)C(=O)OC)CCC1)OC C(=O)(CC(C)C(=O)NCCC1CCCN(C(=O)C(C)(C)c2cncs2)C1)OC CC(C)C(O)C(C)C(=O)NCC1CCN1C(C12CC(CCO1)C2)=O C1(NC(C(C2CCOC2)OCC)=O)(CNC(C2(OC)CCCC2)=O)CCOC1 C12(C(N(C)CC3CCN(C(C4CC(F)(CF)C4)=O)C3)=O)CCC(CC1O)C2 c1(C(N(C(C)C(=O)NCC2(O)CC2)CCC)=O)cn(C(C)C)nn1 N1(C(CCOCCOCC)=O)C2CCC1C(NC(c1c(Cl)n[nH]c1)=O)C2.CC N1(C(C2(OC(C)=O)CC2)=O)CC(C)(NC(c2cnc(O)o2)=O)C1 c1(COC)cccc(C(N2CCC(C)(NC(=O)C(C)CC3CC3)C2)=O)c1 CCC(O)C(C)C(=O)NC1COCCN(c2ncc(Cl)c(O)n2)C1 C(=O)(C(C)CC(F)(F)F)NCC1CN(C(c2cc(C)c(C)nc2)=O)CC1(C)C C=CCC(CC)C(=O)N1CC(OC)C(NC(=O)CCOC2CCCCCC2)C1 C1(Cl)(CNC2CC(NC(C3CCCCC3n3cc(CO)nn3)=O)C2)CC12CCC2 c1(C(=O)NC2C(OC)CN(C(C3(F)CC3C)=O)C2)csc2ccc(F)cc12 C12(OC)CN(C1)C(=O)C1(CC=CC1)CONC2=O.c1(C(=O)NC)ccn(C2CC2)n1 c1(OC)cccc2c1CC(NS(=O)(=O)N(CC(=O)O)C1CCC1)C2 N1(C(CCCCC#C)=O)CC2(CCCC(CNC(=O)CC)O2)C1 C(=O)(C(C)(F)C(C)(C)F)NCc1ccc(C(N(C(C)C(C)(C)C)C)=O)o1 C1(CCC(=O)OCC)CCCCN(C(C)CC(C)(C)OC)C1 c1(C(=O)OC)ccc(NC(C2CN(Cc3cccc(I)c3F)C2)=O)c(Cl)c1 c1(CC)occ(C)c1C(=O)NCC1CC1CNC(=O)C(C)(C)CC1CC1 O=C(CCCCCF)NCCC1CCC(NC(c2cc(C3CC3)ns2)=O)C1 N1(C(c2ccc(-c3ccco3)o2)=O)CC(O)CC1c1cn(-c2nccs2)nn1 N1(C(C(CC)(C)COC)=O)CCCN(C(=O)CC(C)c2cccnc2)CCC1 CC12CN(C(=O)C(=Cc3c[nH]cn3)F)CC1CN(C(C1CC1F)=O)C2 C1(C(N(C)CC2(O)CN(C(C3CCS(=O)(=O)N3)=O)C2)=O)CCC2(CCC2)OC1 C(N=c1nc(Oc2cccc(OC)c2)[nH]o1)c1ccc(OCC)cc1 N1(C(C(COC)O)=O)CCC2(CCN(C(=O)CC3CN(C)C3)CC2)C1 Cn1ccc2c(C(N3CC(NC(=O)CNS(N)(=O)=O)C(O)C3)=O)cccc12 c1(C(=O)NC(CC2CN(C(c3cccc(C)c3N)=O)C2)C)ccc2nn[nH]c2c1 c1(CNC(=O)NC2CC3OCCC23)ccc(-c2ccccc2)c(F)c1 c1(SC)ncc(C(=O)N(C2CN(C(=O)C(C)(C)c3cnco3)CC2O)C)c(O)n1 c1(C(C(=O)NCC(C)CNC(C2C3CCCC23)=O)NC)cccc(C(F)(F)F)c1 c1(CC(=O)N(CCCNC(=O)CC2(C)CC2F)CC)cc(F)ccc1F C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC2(OCC(NC(C(C)n3ccnc3)=O)C2)C1 c1(CN(CC(CC)C(=O)OC(C)C)C)nc(Cl)ccc1Cl CCC(C)(COCC)C(=O)N1CC(C(=O)NCC2(C)CCC2)C(C)C1 Cc1c(N)ccc(C(=O)NC2CN(C(=O)CC3C=CCC3)CC2CC2CC2)c1C c1(C(C(=O)NC2CCC2)N(C)Cc2cc(C3CC3)on2)ccsc1CC C(CC(O)CCc1ccccc1)C1C(C)CCO1.c12nccc(n1)CN1CC2C1 Cc1ccc2snc(C(N3CCC(C)C(CNC(=O)CCC(C)C)C3)=O)c2c1 Cn1cc(Cl)c(C(=O)OC(C)(C)C)n1.C123CC1CN(C2)C(=O)C(=O)NC3 S(=O)(=O)(C(F)(F)F)N1C(C(N2CCC(NC)C2)=O)CCC1 C1(NC(CN(C(c2cccs2)C2CC2)C)=O)COCC1NC(=O)CCc1nc[nH]n1 n1(CCOC)nc(C)c(CNc2cccc(C)c2C)c1C c1(C(=O)NC(CC2CN(C(CCC=CC)=O)C2)C)cc(OC)ccc1Br CC1CN(C(=O)CCNC(=O)CO)CCN1C(C12COC(C1)C2)=O C1(C(N2CCC(CC(=O)N(C(C3(C)CC3)C)C)C2)=O)CC(=O)CC(=O)N1 c1(C(N2CC3=C(CN(C(C(C(C=C)C)C)=O)C3)C2)=O)ccc(S(N)(=O)=O)c(C)c1 CC1(CNC(c2ccccc2F)=O)OCCc2sccc21 C=C1C2C1C(=O)NCCCC1(CC1)NC2=O.c1(C(=O)OC)ccsc1 C1(CNC(C(C(C)C)CN(C)C)=O)CCCC2CN(C(c3cnnn3C)=O)CC12 c1(C2(NC(=O)OC)CCCC2)cccc(Cl)c1.c12nccc(n1)C(=O)N2 C1(NC(C=C2CCC(C)C2)=O)CN(C(=O)CCC(C)(F)F)CC(C)(C)C1 N1(C(C2(CC)CCN(C(=O)CC3OCCC3(C)C)C2)=O)CCc2ccncc2C1 c1(C(=O)NCC(C(C(=O)NC(c2c[nH]ccc2=O)C)F)C)cnc2ccccn12 CCCC(C)(CC)NC(=O)CC1CCCCC1NC(=O)CSC(C)C c1(C(=O)NC)cccc(C(=O)NC(C2CCCN2C(c2cc[nH]c2)=O)C)c1 N1(C(CCC=C)=O)CC(OC)CC1(C)CNC(=O)COCC(C)C C(CC(=O)N1CCOCC(C(=O)O)C1)(C(C)C)OCC.NCC c1(C(N2CC(C=C)C(NC(=O)C(C=C)CC)C2)=O)ccc2c(c1)CCCC2 C(=O)(CCC(F)(F)F)NC1C(N2CCN(CC)CC2)CCC1 Cn1c(=O)c2c(nc(SC3CCC(=O)NC3=O)n2C)n(C)c1=O CCN=c1[nH]c(C(=O)NC2(C3CCCCN3C(=O)C(=O)NCC)CC2)cs1 c1(N2CC(C(C)NC(=O)CCCN3C(=O)CCC3=O)C2)cc(C(N)=O)nc(Cl)n1 N1(C(C(CC(C)C)NC(C)=O)=O)CCC2(CC1)CC(NC(C1(C#N)CC1)=O)CCO2 c1(NCC(CNC(=O)NCC2CCCCO2)F)nc(C2CCCO2)cs1 c1(C(=O)NC2CN(C(C3CCN(C(CC)=O)CC3)=O)C2)cc2n(n1)C(C)CCC2 C1(C(=O)NC2(CC=C)CN(c3ncnc(C)c3Br)C2)CCCCN(C)C1=O CC1C(C(=O)NC2(CNC(c3ccn(C4CC4(F)F)n3)=O)CC2)CCN1C c1(C(=O)NCC(C2CC2)NC(c2c(OC)cc(C)cc2)=O)nc[nH]c2nccc1-2 C1(CNC(C)=O)CCCC(CNC(c2cccc(-n3cncn3)c2)=O)C1 N1(C(c2cc(C3CC3)on2)C(=O)NCCC)CCCCCC1c1ccncc1 C12(NC(c3cnc(COC)s3)=O)CCN(C(C3(COC)CCCCC3)=O)CC1C2 C1(CNC(CNC(N)=O)=O)CCN(C(=O)CSCc2ccncc2)CCC1(F)F C1(F)(CNC(c2cccc(CF)c2)=O)COCCN(C(C2CCCOCC2)=O)C1 c1(C(=O)NC2CC(NC(C3C(OC)CCCC3)=O)C2)n[nH]c2c1CCCC2 C(=O)(C(Cc1ccccc1C)CC)NCC1C(NC(c2ccn(CCC)n2)=O)C1 c1(C(=O)NCC(=O)NC2CCC(SCCC(=O)Nc3ccsc3)C2)ccccc1 N1(C(c2c(C)n(C)nc2)=O)CCCCC1C1CCCN1Cc1c(Br)cnn1C c1(CC)nc2n(n1)CC(NCC(O)COC(C)C)CC2 c1(C(=O)NC2CCC(NC(c3c(C)onc3Cl)=O)C2)cc(O)ccc1Br CCCCC(O)CC(=O)N1CCC2(CC1)CC2CNC(c1cc(OC)ncn1)=O C12(NC(=O)C(F)=C3CCCC3)CC(C1)N(C(=O)CCOc1cccc(Cl)c1)C2 N(C1c2ccc(Br)cc2CC1(C)C)CCN(CCCn1cc(COC)nn1)C N1(C(c2c(C)csc2C)=O)CCOC(C)(CNC(C2CS(=O)(=O)C2)=O)C1 N1(C(c2ccc(C)n2C)=O)CCC12CN(C(C1(C)CC1(F)Cl)=O)C2 c1(C(N(C2CCN(C(=O)C(c3cnn(C)c3)OC)CC2)CC)=O)cccc(=O)o1 C1(NC(c2ccc[n+]([O-])c2)=O)C2CC1N(C(C1(Cl)CC1(F)F)=O)C2 CCC(C)CC(C)C(=O)N1CC2(CNC(=O)COc3ccccc3C)CC1CO2 N(C(=NCCCOc1ccc(C)cn1)NC1CCS(=O)(=O)C1)C(CCCCC)C S(=O)(=O)(c1c(C)noc1C)N1CCN(S(CCOC)(=O)=O)CC1C(C)C c1(C(N(CCCN(C(=O)CCN2CCC(F)C2)C)C)=O)cccc2ccoc12 C(=O)(C1CCCc2ncccc21)N1CCC(C(C)NC(=O)C2=CC3CCCC23)C1 c1(C(=O)NCC2N(C(C(CC(CC)C)C)=O)CC2)cc([N+](=O)[O-])ccc1OC Cc1cc(-c2nc(-c3cnn(C)c3)nn2-c2cccnc2)cc(=O)n1C C1(C(=O)NC(C2CCOCC2)C#C)(NC(=O)CC(O)CC)CCN(C)C1 CC(C)C(C(C)NC(=O)C1=CCSC1)NC(=O)CCc1cccnc1 C1(NC(=O)C=CCN2CCC2)CC(O)C1CC(=O)NC1COCC1C(N)=O c1(NC2CC(C)(C(=O)O)C2)ccc(O)c(OCC(F)(F)F)c1 C1(NC(COCCSC)=O)CC2(CCN(C(C3CN(C)CC(C)O3)=O)CC2)C1 N1(C(c2c(C)scn2)=O)CC(O)CC1(C)C(=O)NCCn1cnnc1 c1(CC(=O)N(C(=O)NCCCCOC)C2CC2)sccc1Br N1(C(c2cnn(C)n2)=O)CCC2CCCC12C(=O)NCCc1ccnn1C N(C1CCCn2cnnc21)C(CCCCCNC(=O)Cc1cccnc1)=O C1(N(C)C)CN(C(=O)CCN(C(=O)CC2CCC(C)(C)O2)C2CC2)CC1O C1(CC(N2CCOC(CF)C2)=O)CC(F)CN1C(=O)Cc1cncnc1 N1(C(=O)CCc2cncs2)CCC2CN(C(c3cnc(C(F)(F)F)nc3)=O)C2C1 C1(CNC(c2scnc2Cl)=O)CC2CCC1N(C(c1c[nH]c(Br)c1)=O)C2 c1(OC)ccccc1C=CC(=O)NC(C)CC(C)NC(=O)Cc1cncc(O)c1 n1(C(C2CCO2)C)cc(-c2cc(CON)no2)nn1 N1(C(C2CCOCC2)=O)CCC(NC(C2(n3cc(Br)cn3)CC2)=O)CC1 N1(C(C2(C)C(C)(C)C2)=O)CCC2(CC1)CN(C(c1ccccc1Cl)=O)CCO2 N1(C(C2CN(C(C(C)C3(O)CCC3)=O)CC(C)C2)=O)CCC(O)CC12CC2 c1(C(=O)NCCC2CC(NC(C3(C(C)(F)F)CC3)=O)C2)snnc1C1CC1 CC1=CCC=CC1C(N1CCCC1CNC(c1cccc(C(N)=O)c1)=O)=O C(CC1CCC2CC12)(C(=O)NCCCSC)N(C(CC#C)C)C.O c1(C(=O)NC2CN(C(c3cc(C)c(F)cc3)=O)CC2O)cc2cncn2c(O)n1 O(N=C1CCCCCC1)CC(=O)N(C1CCN(C(C2(S(N)(=O)=O)CCC2)=O)C1)C c1(OC)ncc(CN(C2(C#N)CCNC2)C(=O)C=Cc2ccc(Cl)cc2)cc1CO S(=O)(=O)(c1ccccc1Cl)Nc1c(C(=O)NCC2(C)CC2)c2c(s1)CCC2 C1(C(=O)NC2(CN(C(C(CC3CC3)OC)=O)C)CC2)Cc2nccn2C1 N1(C(c2ccc(C(C)=O)o2)=O)CCC(NC(C2CCCC(C)C2)=O)C(F)C1 C1(CNC(c2cc(CCO)on2)=O)CN(C(c2cn(C(F)F)cn2)=O)CCCO1 C(=O)(C(C(C)(C)C)NC(=O)CC1CC(=O)NC1=O)NCCN(OC)C N1(CC(N2C(COC(=O)NC)CCCC2)=O)CCOc2cccc(Cl)c2C1 N1(C(COCCCC)=O)CC(=O)NCC1C(=O)NC1CCCCC12CC2 c1(C(N(CC(O)CN(C)C(C2(Cl)C3CCC(=O)C23)=O)C)=O)cnc2occc2c1 CC1(C)CC(NC(=O)CC2CC(F)(F)C2)CN(c2cc(O)ncn2)C1 C=CC1(C=C)COCCN1Cc1nc(C2CCCC2)nn1-c1ccc(Cl)cc1F N1(C(c2cccc(C)c2N)=O)CCC(NC(=O)CC(C)N(C)C)C(C)(C)C1 C12(NC(CCCN(C(=O)OC)C)=O)CCCC1(F)CN(C(=O)COC(F)F)C2 C1(NC(=O)CCn2cccn2)CCCC(C(=O)NCCCc2cccnc2)C1 N1(C(C(Cc2cccc(C)n2)NC(C(C=C)C)=O)=O)CC2C(C1)C2(C)C C1(CC(=O)NCC2CC(NC(C3(CC=C)CCOC3)=O)C2)CCOC1(C)C c1(C(=O)NC2CCC(CCNC(CNC(CC)=O)=O)C2)ccc2cc(C)cn2c1 c1(C(=O)NC2C=CCN(C(C(=Cc3cccs3)C)=O)C2)cncc2nc[nH]c12 CCC(CC)C(C(=O)NCC(O)C(=O)NCC1(CC)CC1)OC C1(C(=O)NCCOCCC#C)C2CC3C(C2NC(=O)CC2(O)CCC2)C13 N1(C(c2cccc(NC(CC)=O)c2)=O)CCCOC(CNC(c2ccsn2)=O)C1 CC1CN(C(=O)CCCN2CCCCC2)CCC1CNC(=O)CCF c1(C(=O)NCCCC(C)NC(C2(CC)CCC(O)CC2)=O)cc(F)cc(C)c1N C=CCC(CNC(=O)C(C)(C)CCC)C(=O)NCC1CCOC1 C1(C(=O)NC2(CNC(C3C(C)OC(=O)N3)=O)CCC2)CCCN2CCCC12 c1(-c2ccc(OC)nc2)cnn2c1CN(C(=O)C(C)Cc1ccccn1)CC2 C(C)(C)(CCC(=O)NC(CN1CCCC1)CC)NC(c1cncc(OC)n1)=O N1(C(C(C2CCCO2)NC(C2CC3CC(=O)C2O3)=O)=O)Cc2cccnc2C1 C#Cc1ccc(C(=O)NCC2(C)CCN(C(=O)C(c3ccncc3C)C)C2)nc1 C1(CCOC)(NC(=O)C(C)C(C)O)CCN(C(=O)CC2CCCNC2=O)C1 c1(C(=O)NC(C2N(C(c3cc(CC)no3)=O)CCC2)C)cn(C)nc1C1CC1 C(=O)(C(F)C(F)(F)F)NCC(CNC(c1c(CC)n(C2CCCC2)nc1)=O)(C)O N1(C(C2CC(C)OC2)=O)CC(C2CCN(C(=O)CC3=CCN(C)CC3)CC2)C1 c1(C(=O)NCC(C)CNC(=O)Cn2cc(CN(C)C)nn2)ccc(N(C)C)nc1 Cc1occc(=O)c1OCC(=O)NCC(C(C)(C)C)NC(=O)C1=COCCO1 C1(NC(C2CCC2)=O)C=CCN(C(c2csc(Cl)c2)=O)C1 CCCCC(C(=O)NCC1(F)CN(C(=O)C=Cc2csnc2C)C1)N(C)C c1(C(=O)NC2C(CNC(CC(CC)SC)=O)CC2)cccc2nccnc12 N1(C(CC(C)C)=O)C2CCCC1CN(C(=O)C(F)(F)CC1CC1)CC2 c1(OC)c(Cl)cc(C(N2CCC(CNC(c3occc3C(C)C)=O)C2)=O)nc1Cl C1(N(C(=O)CCN(CCO)C(C2CC2C(C)(C)C)=O)C)CCCOC1 N1(C(c2[nH]cc(C)c2)=O)CCCCC1C(C)NC(=O)CN1CCS(=O)CC1 C(=O)(CCCS(C)(=O)=O)NCC1C(C)CCN1C(=O)COCc1cccc(F)c1 C#CCC(C)(C)C(=O)NCC1CCN(C(=O)C(C)SC)CC1C c1(C(=O)NC(C)CC2CN(C(=O)CCCN3CCCC3)C2)cnn2c1NCCC2 N1(C(C(CNC(C2CCC(=C)CC2)=O)CC(C)C)=O)CCC2(CC1)CC2C#N C1(C(N(CCN(C(=O)C(O)C2CCCC2)C(C)C)C)=O)CCOC2(CCCC2)C1 CCC(CN(C)C)C(=O)N1CCC(OCCCNC(C2(O)CCOCC2)=O)CC1 c1(C(=O)NC23C(CN(C(CCNC(=O)NC)=O)C2)C3)ccc(CO)c(F)c1 c1(C(=O)NCC2(NC(c3nc(COC)[nH]n3)=O)CCC2)ccc2c(c1)CCCC2 C1(CCNC(C(CC)N(CC)CC)=O)CCN(C(C2CCCC(=O)N2)=O)CC1 CCCCCCCCC(=O)N1CC2(C(N3CC4(CCOCC4)C3)=O)CC1CO2 N1(C(CCC(C)OCC)=O)CC2CCC(C(=O)NCC(C)(O)COC)(C2)C1 c1(C(=O)NC2C(NC(c3n(C)ccn3)=O)CCCC2)sc2ccccc2c1Cl C1(NC(C(COC)N(C)C)=O)CC2CC1CN(C(C1CCC3(CC1)CC3)=O)C2 N(C1CCCc2cccnc21)C(C(N1CCCC(C(=O)NC(CCC)C)C1)=O)=O c1(C2C(C(=O)OC(C(C)C)C(=O)O)C2)ccc2c(c1)OCO2 C(=O)(C#CC(C)(C)CN(C)CC)N(CCCNC(=O)CCCC(=O)NC(C)C)C N1(C(C=C(C)C(F)F)=O)CCN(C(=O)CN2CCN(C)CC2)C2COCC12 c1(C(N2C(CC(=O)N(C(CC)C(=O)OC)C)CC2)=O)c[nH]c2cccnc12 c1(OC)cc(CO)ccc1C(=O)NC(C)(C)CCNC(c1ccc(C2CC2)s1)=O CCCCCCC(C)(CC)C(=O)NCCS(=O)(=O)Cc1cn(-c2nccs2)nn1 C(N=c1[nH]c(N2CCC(C3CNC(=O)C3)C2)nc2c(F)cccc12)C1(SC)CC1 N1(CCN(C)C(C23CCCC2CC3)=O)CCN(C(c2cc(Br)n(C)c2)=O)CC1 N1(C(c2cc(C#N)sc2)=O)CCN(C(=O)Cc2cccc(F)c2)C2CC12 N1(C(c2ncc(C(=O)OC)s2)C(=O)NCCSC)CC(CCO)OCC1(C)C CCC(CC(F)(F)F)NC(C12C(NC(=O)Cn3[nH]cnc3=N)C3CC1C2C3)=O n1(CC)nc(C(=O)NCC(C2CC2)N(C(=O)C(C)(C)c2ccn(C)n2)C)c(C)n1 CC1CCCC(O)(C(=O)Nc2csnc2C(=O)O)CC1 N1(C(C(C)=O)=O)CCC2(CC1)CC2NC(c1cc(C)ccc1F)=O CCCCCCC(C)(C)C(=O)NC1CN(C(c2ccnn2CCOC)=O)CC1O C1(C(=O)Nc2ccccc2Cl)C2Cc3ccccc3C12.CCC1CNC(=O)CO1 c1(C(N(C)CC2CCCN(C(c3cc(CCC)[nH]n3)=O)C2)=O)cn2c(n1)SCC2 C1(CC(=O)NCC(CNC(CCOCCCC)=O)C)(N(C)C(=O)OC)CCCC1 c1(OC)ccc(OC)c(C(=O)NC2CCN(C(=O)CS(N)(=O)=O)C2)c1OC C1(CC(=O)OC)C(=O)N(C)CCN1Cc1ccc(OC)c(C#N)c1 N1(C(CC(C)N(C)C)=O)CCCCC(NC(=O)CC2CCN(C)C2)C1 c1(CN(CC(=O)N(CC(C)NC(C)C(=O)Nc2cnn(C)n2)C)C)ccccc1 CC(C)C(CCNC(=O)CC1CCC(C)C1)NC(=O)C=Cc1cnc[nH]1 C1(C(=O)NC2CCCC2(C)CN(C(=O)C(C)(C)C)C)(COC)CCOCC1 c1(C(=O)NC(Cn2cc(C(=O)OC)nn2)C)cc(C(F)(F)F)cc(F)c1 c1(CC(=O)NCCCC2CCCN2C(=O)CSC(F)F)cccc(O)c1 c1(N2C(=O)CCC2)ccc(-n2ccnn2)c(Br)c1.C12CC(=O)N(C(=O)N1)CC2 C(=O)(C(CO)C(F)(F)F)N(C)CC1N(C(Cc2ccc(C)o2)=O)CCCC1 N1(C(CCC(CC)C)=O)CC(C(=O)NCCC2(CO)CC2)C2(CCC2)C1 n1(CCN(CCOC)C(c2ccccc2)=O)sc2ccccc2c1=O N1(C(C(C)NC(CC)=O)=O)CCN(C(=O)COc2ccc(C)cc2C)CC1CO c1(C(=O)NCCNC(=O)C(C2CC2)NC(c2ccnnc2)=O)ccnc(CO)c1 c1(COCC)nnc(COC(C2(C)CC(C(=O)OC)C2)=O)o1 N1(C(CCCC)(C)c2nnnn2C)CCS(=O)(=O)C2(CCC2)C1.C1(O)CN(C(C)=O)C1 N1(C(C)=O)CC(C(=O)NC2CCOCC2)C2(C1)CN(CCC(C)F)C2 C1(C#CC(=O)NC2CC3CCC(C2)N3C(=O)C=C2CCC(C)CC2)(CC)COC1 C(=O)(C(C)CCCc1ccccc1)N1CCCC(N(C(c2cnns2)=O)CC)C1 N1(C(c2cncn(C)c2=O)=O)CC2CN(C(c3ccccc3Cl)=O)CC2(C)C1 c1(C(=O)NCC(CNC(c2c(SC)scc2)=O)C)cccc(C#N)c1 C=CC(C)(O)CC(=O)N1CCC(NC(=O)COc2ccc(C)cc2C)CC1 c1(C(=O)NC2CC(NC(C3(N(C)C)CC3)=O)C2)cnccn1 CC1CN(C(C2(C)CCN(C)CC2)=O)CCC1CNC(=O)C(F)(F)c1nccs1 N1(C(C(C)OCC#C)=O)CCCCC1C1(NC(c2cc(CO)n(C)n2)=O)CC1 N1(C(CCOCC#C)=O)CCN(C(C23CCCC2(C(=O)OC)C3)=O)CC1CO C12(NC(CCC=C)=O)CCC(CC1NC(C1CC(C)(C(C)(C)C)C1)=O)C2 CC(C)(C(=O)N1CC2CC(NC(c3csc(-c4cn[nH]c4)n3)=O)C2C1)C(N)=O c1(OC)cc(CN2CCN(C(=O)CCNC3(Br)CCC3)CC2)cc(OC)c1OC n1(CC)nc(C)c(C(=O)NC2CS(=O)(=O)CC2NC(c2ccc(C)cn2)=O)c1C c1(CNC(C(C2CC2)SC)=O)cn(C(C)C(=O)N2CCCC2)nn1.c12ccoc1C2 CC1(CNC(C2(CO)CCCO2)=O)CCCN(C(=O)Cc2cc(F)ccc2Cl)C1 CCCCCCCC1CCCN1C(c1cnn(C2CC2)c1)C(=O)NCCCSC n1(CC)nccc1C(N1CCCC1CCCNC(=O)CNc1ccsc1)=O c1(C(N(CCC)CCNC(=O)C(CC)N(C)C)=O)cc(S(N)(=O)=O)c[nH]1 c1(C(=O)NC23CC(C2)N(C(c2cncnc2)=O)C3)c(C(F)F)nc2ccccn12 C1(CC(=O)NC2CN(C(CC)=O)C2)CCCCN1C(C1CC(C)=NO1)=O c1(C(N2CC(CCNC(CC(C)(C)OC)=O)(OC)C2)=O)cnc2n(c1=O)CCS2 N1(C(C(c2ccc(C)s2)C)=O)C2CCC1CC(CNC(=O)Cc1sccc1C)C2 N1(C(c2cc(C)n(C)c2)=O)CCCC(C)(CNC(C2(O)COC2)=O)C1 c1(OC)cc(Cl)ccc1C(=O)NC1CC(NC(=O)CN(C)C)C12CCC2 c1(OC)cc(OC)nc(C(N2CCN(C(C3CCCCCC3)=O)CC2)=O)n1 CC1CC2(CC2)CN1C(=O)CC(CC1CC1)NC(=O)C(=O)NCC1CC1 c1(C(=O)NC(C2(O)CN(C(CCOC(CC(C)C)C)=O)C2)C)ccc(Cl)c(F)c1 CCC(CC(=O)N1CCC(CNC(c2nnc(O)cc2O)=O)CC1)C(C)(C)C c1(C(N2CCC(C3CC3)C2)C(=O)NC(CC)C)ncc2ccccn12 CCCCCC(C)(CC)C(=O)NCC1(O)CC(CNC(C2(SCC)CCC2)=O)C1 Cc1cccc(NC(C2COC(CNC(=O)CC(F)F)C2)=O)c1 c1(CC(N2CC(F)(C(=O)NCC=Cc3ccco3)C2)=O)ccc(Br)cc1 C1(C(=O)NCC2(NC(C3CCCCO3)=O)CCCCCC2)CS(=O)(=O)CC12CC2 Cc1ccc(CCC(=O)N(C)CC2CCCN2C(C2CCCC(O)C2)=O)c(C)c1 C1(CC(=O)NCC2(CNC(C3(C)CC(=C)C3)=O)CC23CCC3)NC(=O)CNC1=O c1(CNC(CN(C(C)=O)C)=O)cccc(CN(C)C(c2n[nH]c(O)n2)=O)c1 C1(C(N2CCC(NC(c3cc(O)ncn3)=O)C2)=O)Cc2cccnc2C1 N1(C(C(CC)(C)COC)=O)CC2CCCN(C(c3n[nH]c(C)c3C)=O)C2C1 n1(CC(=O)NCC2CN(C(Cc3c(C)non3)=O)C(C)C2)cc(Br)ccc1=O N1(C(C2C(CNC(C3CN(C(C)=O)C3)=O)CC2)=O)CC(=O)N2CCCC2C1 c1(CC(N2CC3(CN(C(c4c(C)cc(N)cc4)=O)C3)C2)=O)cn2ccccc2n1 c1(C(=O)NC(CCCC)CNC(c2cc3n(n2)CCC3)=O)ncnc2cc[nH]c12 c12cccc3nc([nH]c13)CC1CN(CCO1)C(=O)N(C)C2.C(C)(C)(C)O C12(CNC(C(CC=C)OC)=O)CCC(CN(C(C3(OCC)CCC3)=O)C1)C2 C=C1CCN(C(c2cnnc(C)c2)=O)C(C(=O)NCc2cn(C3CC3)nn2)C1 N1(C(c2ccoc2)=O)CCN(C(C2C3CNC(=O)C23)=O)C2COCC12.O=C1CN1 C(=O)(C1=NNC(=O)CC1)N1CCC(C)(C)C1CNC(=O)CC1CCCOC1 c1(C(C(=O)NCCC2(O)CN(C(c3ccc(=N)[nH]n3)=O)C2)O)cc(F)cc(F)c1 C1(C(=O)NCCCOCC#C)(OC)CCC(C)C1.C12CCCC1C(=O)N2 c1(C(=O)NC(C2CCN(C(C3(CO)CC(F)(F)C3)=O)CC2)C)ccc(CO)cc1 C(=O)(C#CC1CCCO1)NC1(CF)CCN(C(c2c(C)ocn2)=O)C1 N1(C(C2C(C(=O)OCC)CC2)=O)CCCCC(NC(C2CCN(C)CC2)=O)C1 CCCC(C(O)C(=O)NC1CCCCCCC1O)NC(=O)C(C)CC(C)(C)C c1(N(C2CCN(c3nc(OC)c(C)cn3)C2)C)ncc2ccc(Br)cc2n1 C(=O)(CC(C)(C)C(F)F)NCC(CC(=O)NCc1nccc(C)n1)(C)C C12(OC)CCC(C(=O)NCCC3CN(C(c4cnc(C)n4C)=O)CCO3)(CC1)C2 c1(OC)noc(C)c1C(=O)NCc1ccccc1CN(C)C(c1ncn(C)n1)=O N1(C(C2N(C(CCOCC)=O)CC=C2)=O)CCCOC(C(C)C)C1 c1(C(N2CC=CCC2(C)C)C(=O)NCCSC)cc2ncc(Br)cc2o1 c1(C(ONC(=O)NCC2CCN(c3ccncc3)C2)C)cnn(C)c1F C1(N(C)C(C2C3COCC23)=O)CN(C(=O)CC2CC(=O)NC(=O)C2)CC12CCC2 Cc1occc(=O)c1OCC(=O)NC1(CNC(C2C(C=C(C)C)C2(C)C)=O)CC1 C1(NC(CCCNC(c2cc(C)[nH]c2C)=O)=O)CCC2CCCC1O2 N1(C(C(C=C)O)=O)CCCC2(C1)C(NC(=O)CCCCCC(C)C)CCN2C C1(NC(c2cc(CC)n(C)n2)=O)CS(=O)(=O)CC1N=c1ccnc(C(C)(C)C)[nH]1 Cc1cc(C(=O)N(C2CN(C(c3ccnn(C)c3=O)=O)CC2F)C)c(C)cc1Cl c1(OCC(=O)NC(CCOC)CNC(c2c[nH]nc2Cl)=O)ccc(F)cc1 C#Cc1ccc(NC(=O)CC2CCN(C(=O)OC(C)(C)C)CC2)c(Br)c1 n1(C(C(=O)NC(CCNC(c2cnc(C(C)=O)s2)=O)C)C)cnc(C#N)n1 c1(CNC(CCN(CC#C)C(c2ccns2)=O)=O)cc(C)c(C)s1 C12(C(=O)NCC3CC(NC(c4n(C(CC)C)ncc4)=O)C3)CCC(C1)C(C)(C)O2 C1(CC)CCOC1C(=O)NCc1csc(CNC(=O)CN(c2cnccn2)C)n1 c1(CN(C(=O)C(=O)NC2CCCC23CCC3)C)ccc(OC(F)F)cc1OC(F)F CC(CC(=O)N(C)CC1CCC(NC(=O)CN(C2CCCC2)C)CC1)C(C)(C)C C1(NC(c2ccc(-c3ccc(C)s3)s2)=O)CC2CC1N(C(C1CS(=O)(=O)C1)=O)C2 CC(C)(C(=O)O)n1cc(CCNC(=O)Cc2ccc(Cl)s2)nn1 C(C1CCCN1C)=CC(N1C(C(C)(C)NC(C(C2CCOCC2)C)=O)CCC1)=O C(=O)(C1=C(Cl)CCCC1)NC(C1(O)CCN(C(c2c(C)n(C)nc2Cl)=O)CC1)C C1(C(CN)C(=O)NC(c2ccccc2)Cc2ccncc2)CCCCCC1 c1(C(=O)NCC(CCOC)NC(=O)COc2cccnc2)c(C)n[nH]c1C N1(C(C2C(CC)OCC2)=O)CCN(C(C2COCCN2CC(F)F)=O)CC1CO c1(C(=O)NCC(CCNC(C2CC2C2CCOCC2)=O)O)cnn2ccccc12 c1(N2CC(CNC(c3c(CC)ocn3)=O)N(C)CC2)c(C)cccc1[N+](=O)[O-] N1(C(c2cc(C)nn2C)=O)CCC(NC(=O)COCc2ncnn2C)C(CO)C1 c1(OC)nc(C(=O)NCC(C2(C)CC2)NC(=O)OC(C)(C)C)co1 C1(CNC(c2cc(C)oc2)=O)CC(O)CN1C(C1CC2(CC2)CO1)=O C(=O)(C1CCCc2sc(=N)[nH]c21)NC1CC(NC(c2c(CC)ccc(F)c2)=O)C1 O=C1CCCc2cccc(NC(C3(F)CN(C(C4CCC4)=O)C3)=O)c21 c1(C(N2CC3CCN(C(C(CSC)C)=O)CC32)=O)cc(C)cc2c1CCC2 CCC(CC)C(C)C(=O)N1CC(C2CN(C(C3CCCC(C)(C)O3)=O)C2)C1 C(=O)(C(C)S(N)(=O)=O)NCC(CCCC)NC(c1ccc(C2CC2)nc1O)=O C(c1cnn(-c2ccccc2)c1)=CC(=O)NCCCCN(C)C(c1cscn1)=O N1(C(Cc2c(C)cccc2)=O)CC2CCC1C2NC(c1ccc(O)c(CO)c1)=O N1(C(C(CC)(C)C#N)=O)CC(C(=O)NC(c2cccc(SC)c2)C)CC(C)(C)C1 C(=O)(CCCCN1CCCCC1)NCCC(C)NC(c1nnc(C(C)(C)C)o1)=O C1(C(=O)NC(C(=O)NC2(CC=C)CCC2)C2CCCO2)CC(=O)OC1(C)C C1(CC(N2CC(CC(C)NC(c3ccccc3CO)=O)C2)=O)CN2CCN1CC2 c1(C(N2CC3(CC(NC(C(C)NC(=O)NC)=O)C3)C2)=O)cccc2[nH]c(C)cc12 C#CCC(C(=O)NC(CC)C(C)(C)O)NC(=O)CCn1cnc(=N)[nH]1 N1(C(c2ccc(NS(=O)(=O)C3CC3)cc2)=O)CCC2CCNCC12 Cc1csc(=NCC(=O)NC(C2CCN(C(=O)CCC3CC3(Cl)Cl)CC2)C)[nH]1 c1(OCC(=O)NC2C(NC(C(C(C)C)=O)=O)COCC2)ccc2ccccc2c1 c1(OC)ccc(C2(C(=O)NCCN(C(C)=O)C3CC3)CC2)cc1.N1CCCCC1 S(=O)(=O)(C1(c2cn(C(C)C(N3CCCC3C(F)(F)F)=O)nn2)CC1)NC C1(NC(C2C(C(=O)OC)C=C2)=O)CN(CC2CCOC2(C)C)C2(CCCCC2)C1 C1(NC(c2[nH]ccc2C2CC2)=O)CC(NC(C2CCCOCC2)=O)C(O)C1 N1(C(C(C)=C(CC)C)=O)CCC(CNC(c2ccc(C(F)F)o2)=O)(OC)CC1 C1(CC)CCN(C(=O)Cc2cnn(C)c2C)C1CNC(c1ccnc(OC)n1)=O CCC(COC)(CC)C(=O)NC1CCCC(NC(c2ncncc2C)=O)C1 C1(CNC(CCN(C(CC)CC)C)=O)CC(O)CN1C(c1ncoc1C)=O N1(C(C(CC)C(F)(F)F)=O)CC2CCC(C1)C(NC(c1cc(OC)nn1C)=O)C2 Cc1cnc(S(C)(=O)=O)nc1N1CCC(C(=O)NCc2ncc(Br)s2)C(O)C1 N1(C(C(C)OC2COC2)=O)CC(NC(C2(CO)CCC2)=O)CCC1C C1(NC(CC(C=C)CC)=O)C2CC3CN(C(c4snnc4C)=O)C1C3C2 C1(NC(c2cccc(N(C)C)n2)=O)CN(C(C2CCS(=O)(=O)C2)=O)C(C)(C)C1 c1(OCC(=O)NC2CCCC2NC(C2CC3CCC3C2)=O)ccc(F)nc1 C=C(C)CN=C(NCC(C)(C)OC)NCC(c1ccc(F)cc1)(C)C N1(CCC2(C(=O)NCCN(C)C(=O)OC(C)(C)C)CCCC2)CCC(CO)CC1 CCC(F)(F)C(=O)NCCC1CN(C(c2conc2C(C)C)=O)CCO1 c1(N2CCOCC(NC(C3(N(C)C)CCCCC3)=O)C2)nc2ncc(Cl)cc2o1 C#CC1(O)CC(C(N2CCN(CCCNC(c3nc(Cl)sc3C)=O)CC2)=O)C1 c1(OC)n[nH]c(=NC(=O)C(Cc2ccccc2)NC(c2ccccc2)=O)s1 c1(CN2CCC(C#N)(NC(C3(C#N)CCC3)=O)C2)cc(F)c(O)c(F)c1 Cc1cc(C)n(CC(C)NCC(=O)Nc2ccccc2N2CCOCC2)n1 c1(C(=O)NC2CCN(Cc3c(OCC)cccc3)C(C)C2)ccc(C#N)cc1O N1(C(CCC2C(C)C2)=O)CC(CO)C2(C1)CN(C(=O)CCC1CCCCC1)C2 Cc1cc(Cl)cc(NC(C2CN(C(c3cccc([N+](=O)[O-])c3)=O)CCS2)=O)c1Cl N1(C(CCOCCN(C(=O)Cc2ccc(O)cc2)C)=O)CC2CCN(C)C2C1 N1(c2nnc(CCOC)s2)CCC2CC(NC(=O)CC3C=CCCC3)CCC2C1 C(C(F)(F)C(=O)N(C1CC2(CNC2)C1)C(C)C)OCc1ccccc1 CC1=C(C(=O)N(CCCNC(c2n[nH]c3cccnc23)=O)C2CC2)CCCO1 C1(CNC(C2CCC(OC)CC2)=O)CN(C(=O)C(C)OC)CCC1(F)F c1(NC(C2CCN(c3nnnn3C(C)(CC)C(F)(F)F)C2C)C)cccc(=O)n1C C=CCC(F)(F)C(=O)N1CC(NC(=O)CC2(OC)CCCCC2)C(C)(C)C1 N1(C(C(CC)OCC)=O)CCCN(C(=O)C=C(C)c2ccccc2)C(C(C)C)C1 c1(C(=O)NC(CNC(COCC)=O)(C)C)cnn(CC(F)F)c1 N#CCCCCC(=O)N1CCC(OCCNC(c2ncccc2N(F)F)=O)CC1 N1(CC=C)CCN(C2CCN(C(=O)CCOCCOC)C2)CC1 C1(NC(CC=CC=C)=O)CCN(CC2(C(=O)NC)CCC2)C1 Cc1ccc(C=CC(=O)NCC2CN(C(=O)CNS(=O)(=O)N(C)C)CC2O)cc1 C(=O)(CC(C)n1cccn1)NCCCN(C(=O)C(O)C1CCC1)CCC N1(C(C2N(C(CCC(C)(F)F)=O)CC=CC2)=O)CCC12CCSCC2 c1(CC)c(OC)cccc1C(N1CCC(NC(C2CC2(F)F)=O)C(F)C1)=O CC1CC(CO)CN1C(=O)Cn1cc(CNC(=O)CC(Cl)Cl)nn1 C=CCC(C(=O)NC(C)(CNC(=O)COc1ccccc1C)CC)NC(C)=O N1(C(CCN(C(=O)COCC2CCCOC2)C)=O)CCN(C)C2(CC2)C1 CC1CN(C(=O)Cc2ccc(Cl)cc2)CC1NC(C1(c2cccs2)CC1)=O c1(C(=O)NC2CN(C(c3ccco3)=O)CC3C2C3)cccc2c1COCCN2 N1(C(CC(CC)O)=O)CCCCC(C(=O)NC(C2CCCCC2)C)C1 C1(NC(COC(CC)C)=O)CCCCC1CNC(c1ncccc1CC1CC1)=O C(=O)(CC(C)C(C)(C)C)NC(C1N(C(CCCNC(=O)OC)=O)CCC1)C N1(C(c2ncc(C)cc2F)=O)C2CCC1CN(C(c1ccc(F)s1)=O)C2 N1(C(C2CC(OCC)C2)=O)CCOCC(NC(C2(C(F)(F)F)CCC2)=O)C1 c1(CN2CC(F)(C(=O)NC(CCSC)CO)C2)c(F)c(F)cc(F)c1F C1(NC(=O)COc2ccccc2O)CCCCCN(C(=O)Cc2ccoc2)C1 C1(c2n(C)nnn2)(NCC(=O)Nc2ccccc2C2CC2)CCN2CCCC12 C1(NC(C2ON=C(C)C2)=O)CCC(NC(=O)Cc2cc(Cl)cs2)CC1 N1(C(C2CC(SC)C2)=O)CC(NC(c2cc3cn[nH]c3cn2)=O)CC12CCOC2 N1(C(c2c(CC)nc(C)[nH]2)=O)CC(CNC(=O)CCC2CCOCC2)CCC1C Cc1ncccc1CNC(c1ccc(CNC(=O)Cc2ccns2)nc1)=O C=C(CNC(c1ccc(C(C)C)o1)=O)CCNC(=O)CN1CC=CC1 C(=O)(C1=NN2CCCN=C2N1)N1C2CCN(C(C3C=C(C)CS3)=O)CC2CC1 C(=O)(CC(C(C)C)OCC)NC1(CNC(C=CC)=O)CCOC1 c1(COC)nc(C)cc(=NC(=O)c2cc(C(F)(F)F)cc(N)c2)[nH]1 CCCC(C(=O)NC1CCC1C(=O)OC)NC(c1ccc(OC)o1)=O N1(C(c2cc(CC)[nH]n2)=O)CCN(C(C2(C)CCCS2)=O)CC1C1CC1 C(=O)(C1CCc2cccc(F)c21)N1CCC(C(C)NC(C2CNC(=O)C2)=O)CC1 N1(C(CNC(N)=O)=O)CC2CN(C(C3C4COCC34)=O)CCC12 c1(C(=O)NC2C(CNC(c3ccc(OC)c(F)c3)=O)C2)cccc2scnc12 C(=O)(C(O)C(C)(C)C)NC1C(C)(CNC(c2ncc(CC)cn2)=O)CCC1 C(=O)(C(C#N)C(C)(C)C)NC1CCCC(C(=O)NCCOC(CC)CC)C1 c1(OC)ccc(CC(N2CCC3CC23C(=O)N(C)CC2CCN(C)C2)=O)cn1 C#CCC(CC(F)F)C(=O)NCC1CC1CNC(C1NC(=O)OC1C)=O N1(C(CC(C=C)C)=O)C(C)CC2CN(C(c3coc(C4CC4)n3)=O)CC12 C(=O)(CCCC(C)(C)CC)N(CC(C)C(=O)NC)Cc1ccc(CCC)cc1 n1(C(C)C)ccc(CNC(C2CC2C(=O)Nc2cn(CCN(C)C)nn2)=O)n1 c1(C(N(C2CCN(C(CSCC=C)=O)CC2C)C)=O)cnc2ncccc2c1 C(C(C(=O)NC1CCCC1N(C)C)n1cc(CCCCO)nn1)OCC c1(C(N2CCCC(CNC(c3cnc(C)o3)=O)C2)=O)ccc2c(c1)N(C)CCO2 C1(C(N2C(COC)C=CC2)=O)CNC(=O)CN1C(c1[nH]ccc1COC)=O C1(CNC(C=CC)=O)CCN(C(=O)CNC(=O)CCCCC)C(C)C1 C1(CCN(C)C)CCN(C(=O)C(=O)NCC2CN(C(=O)NN(C)C)C2)CC1.NC Cc1[nH]nc(C(N2CCCC(N(C(=O)CCNC(c3ccco3)=O)C)C2)=O)c1O C1(NC(c2ccc(Cl)cn2)=O)CCCN(C(=O)C(c2ccccc2)C2CC2)CC1 C1(NC(CC(c2ccc(CC)cc2)C)=O)CC2CN(C(=O)C=C(C)C3CC3)CC12 C1(C(=O)NCC2(O)CN(C(=O)CCc3cncnc3)C2)(SC)CC(O)C1 c1(SC)c(C(=O)NCCC2CCN(C(=O)CC3COCCO3)C2)cnn1C Cc1ccc2ncc(C(=O)NCC3(F)CCN(C(=O)C(C)C(C)(C)C)C3)n2c1 N1(Cc2nn(C)c(C(F)F)c2)CC(NC(C2CC(=O)N2)=O)CC2(CCOCC2)C1 C1(C(=O)Nc2cnc(C)c(Cl)c2)CCCC12CCN(C(=O)Cc1cc[nH]n1)C2 C1(CC)(CC)CC(NC(c2ccnc(C)c2)=O)CN1C(c1ccoc1)=O C(CC(C)(C)CNC(C1CC2CCC1O2)=O)NC(CCOCCC)=O C(=O)(CCC(=O)c1ccccn1)NCC(CNC(c1c(COC)nn[nH]1)=O)(C)C C#CC(CNC(C1CC(NC(=O)COCC(=O)NCCO)C1)=O)CSC n1(CCC)ncc(C(=O)NC2COCC2NC(=O)C(c2c(C)n[nH]c2C)C)c1C C1(C)(C(=O)NCc2nc(CNC(CC(C)C)=O)sc2)CC2CCC(C1)S2 CCC(C)(C)C(O)C(=O)N1CCCC(C)(CNC(c2cccc3ncsc23)=O)C1 c1(C(N2CCC(F)(C(=O)NCC(c3ccccc3)O)C2)=O)ccc(F)cc1Br C#CCC(C)(C(=O)NCCn1cccn1)NC(=O)CC1CCCCCC1 CCCCC(C(=O)N1CC(NC(=O)CN2CCCC2)C(C(F)F)C1)NC(N)=O CCC(CCC(=O)NC(c1nccc(C)n1)C)NC(c1cc[nH]c(=NC)c1)=O C1(CC)CN(C(c2coc(N(C)C)n2)=O)CCC1NC(=O)CCOCC(F)(F)F C12(CNC(c3ccccc3Oc3ccc(Cl)cc3)=O)CCC(CC1O)C2 C(=O)(C1=C(C)CC(C)(C)CC1)N1CC2C(NC(c3cnc(CC)[nH]3)=O)(C2)C1 c1(C(=O)O)cc(CNc2cnc(-c3ncccn3)s2)on1 c1(C(=O)NC(C2CCN(C(C(C)OCCC=C)=O)C2)(C)C)ccc2cc[nH]c2c1 N1(C(=O)Nc2c(C)cco2)CCCc2c(Br)ccc(Br)c21 C(=O)(CCCC(=O)NC(C)C)NCC(CNC(c1cncc(C)c1)=O)O N1(C(C)=O)CCc2ccccc2C1CC(=O)NCc1cnc(O)c(F)c1 N1(C(C(CC(=C)C)C)=O)CCC2CCN(C(=O)CCCn3cccn3)CC12 S(=O)(=O)(c1cc(Cl)cc(Cl)c1O)N1CCN(S(CCC)(=O)=O)CC1C(F)(F)F c1(NC2(c3n(C(CC)(C)C)nnn3)CSCC2C)ccc2[nH]nc(Cl)c2c1 CCC(C(C)(C)O)NC(C1CN(C(c2ccnc(C)c2)=O)CC1C)=O c1(SCCCC)cccc(C(N2CCC2CNC(=O)C(C)(C)Br)=O)c1 C(C(C)C(=O)N(C)C)(c1ccccc1)NCC(=O)Nc1ncc(C)s1 N1(C(Cc2ccc(C)cc2)=O)CC(C2CN(C(c3cncnc3C3CC3)=O)C2)C1 C1(NC(C(C)NC(=O)NC)=O)CC2(CCN(C(=O)CC(O)CCC)CC2)C1 c1(OC)ccc(-c2ccc(CNC(=O)C(C)SC)nc2)cc1O Cc1ccc(Cl)cc1N1CC(c2nnc(CN(C)C)o2)CC1=O C(C)(C(=O)NCC1(C)CCN(C(=O)C2=CCCOC2)C1)(C(C)C)NC(C)=O C(=O)(C1=CCS(=O)(=O)C1)NC1C2(NC(COCc3cc(C)on3)=O)CCC(C1)C2 C(C(=O)N(C)CCNC(=O)C=CCF)(c1cccs1)SC C12(NC(CSC)=O)CC(CSC3CN(C(=O)COC(F)F)C3)(C1)C2 N1(C(C2CCCC(C#N)C2)=O)CC2(CCN(C(=O)CCn3cnnn3)CC2)C1 C1(C)(NC(C2CC(C)(C)C2)=O)CCN(C(=O)C(F)(Cl)c2ccccc2)C1 CC1CN(C(c2ccc(Br)cc2)=O)CCCN1C(=O)COC(F)(F)F C1(CNC(COCC=C)=O)CN(C(=O)C(CC)NC(N)=O)CC12CC2 c1(C(N2CCC(C(F)(F)F)(OC)C2)C(=O)NCCCSC)cc(F)ccc1F C1(CCC)CN(C(C2(c3ccccc3Cl)CC2)=O)CCN1C(C1CCCOC1)=O c1(CN(CC(COCC#C)O)CC2CCCC2)ccccc1F N1(C(C2CCC(=C)CC2)=O)CCC2CCCN(C(=O)C=CC3CC3)C2C1 N1(C(C(C)NC2N(C(C)=O)CCC2)=O)CCC(CN(c2cc(C)ncn2)C)CC1 FC1(F)CCC(n2nc(-c3ccsc3)nc2C)CC1.n1(C2CC2)ccnn1 CC1C(=O)N(CC(=O)NC2CN(C(c3cn(C)c(O)n3)=O)CC2(C)C)C(=O)C1C C(=O)(C(O)C(C)(C)C)NC(C)CC1CN(C(C2(CC3CCC3)CC2)=O)C1 c1(C(N(C2CC(NC(c3c(N)ccc(C)c3)=O)C2)C)=O)cccc2ncn(C)c12 N1(C(c2ncc(OC)cn2)=O)CCCC2(C1)CN(C(=O)C(c1ccc(C)o1)C)C2 C=CCC(CNC(C1(C)CCCO1)=O)NC(=O)C(F)=C(C)C1CC1 Cc1cc2c(cc1C)C(C(=O)N(C1CCCN(C(C3(C)CC3C)=O)C1)C)CO2 C=CCC(C)(CC=C)NC(C1(CNC(=O)CC2CCSCC2)CC12CCC2)=O C1(C(=O)NCC2CCCCC2NC(C2(O)CC2)=O)CC2(C1)CC1(CC1)C2 CS(=O)(=O)CCC(=O)NCC1=CCCN(C(C2CC=CC(O)C2)=O)C1 CCC(C)(CNC(c1cc(C)nnc1C)=O)C(=O)N1CCCC(CCO)C1 c1(CC(=O)NC2CC(CCNC(=O)CCC3CCCCO3)C2)c(F)cccc1Cl Cc1ccc(Cl)cc1CCc1nc(-c2cccnc2O)nn1-c1cccc(Cl)c1 N1(CC)CC(C)c2ccc(S(=O)(=O)N3CCOC(C4CC4)C3)cc21 CC(C)S(=O)(=O)CC(=O)N1CC2CC1CC2NC(=O)CSCc1ncc[nH]1 C1(C(=O)NC2CCN(C(C3CCS(=O)(=O)N3)=O)C23CC3)CC2(C1)CS(=O)(=O)C2 CC(C)CC(F)C(=O)N1CCCCC1c1cn(CCC(=O)CCCCC#N)nn1 N1(C(COC)=O)CC(C2CCCN(C(c3ccccc3OCCF)=O)C2)C1 c1(SCC)cccc(N(C(=O)C(C2CCOCC2)OC=O)C)c1.C1(O)CCCOC1 c1(OC)cc(N)ccc1C(N1CC(=C(F)CNC(C2CNC(=O)N2C)=O)C1)=O C1(C(=O)NCc2c(C)noc2C)CN(C(=O)CC2CC3(CC3)CO2)CCC1(C)C C#CCC(C)(CNC(C1CCCCN1C(=O)CCCC(=O)OCC)=O)CO N(C(=NCC1(c2ccccc2)CC1)N1CCS(=O)(=O)CC1)CC(C)(C)C C(=O)(CC(CC(C)C)NC(=O)COC1CCCC1)NCC(CO)OC.OCC c1(C(C)(F)F)cccc(C(N2CCC(F)(CNC(c3cc(CN)no3)=O)C2)=O)c1 C1(CNC(c2c(CCC)cccc2)=O)CN(C(=O)C(C)C2CC2)CC(C)(C)O1 C1(NC(C(C)NC(=O)Cn2cnnn2)=O)CC2CC(NC(=O)C3CC3)CC12 c1(OC)cccc(SCC(N2CC(CNC(=O)C(F)=C(C)C3CC3)CC2C)=O)c1 N1(C(C(n2ccc(C)n2)C)=O)CC(C#N)(C#N)C1 C(=O)(CCCCC1CC1)NCCC1CCC(NC(CSCC)=O)C1 C1(CNC(C2C(C)OC(C)C2)=O)CC(N=c2[nH]c3ccc(O)cc3s2)C1 N1(C(C(C(C)C)CNC(=O)COCC2CCOC2)=O)CC2(C)CCC2(C)C1 C1(CN(C(=O)C(C)N2CCCC2)CC)CCCN1C(c1ncoc1C)=O c1(C(=O)NC(CN(C(c2nn(C)cc2C)=O)CC)C)nc(C)n2c1CCCC2 c1(CC(=O)N(C2CCCN(C(=O)C(O)CC(N)=O)CC2)CC)ccc(C)c(C)c1 c1(C(=O)NC(C#C)CC(C)C)cc(Br)cc2nc[nH]c12 C1(NC(c2cnc(C(C)C)[nH]2)=O)C(C)CN(C(=O)CC2(CN(C)C)CC2)CC1C CC(C)CC(=O)C(=O)NCCC1(C(=O)NCC2(O)CCCOC2)CC1 N1(C(Cc2c(C)noc2C)=O)CC2CC1CN(C(C1(C)CCCN1C)=O)C2 Cc1ccc(-n2nc(-c3ccncc3)nc2CCN2CCOCC2)cc1C C1(NC(C(CC)n2cncn2)=O)CCC(O)CN(C(=O)CCc2cnoc2)C1 c1(OC(C)C(=O)NC(C)CN(C)C(c2cc(Br)co2)=O)ccc(F)cc1 CCC(CC(=O)N1CC2CC1C2CNC(=O)Cc1cnn(C(C)(C)C)c1)C(C)C S(=O)(=O)(c1c[nH]ccc1=NCCc1ccc(Cl)cc1)NC1(CCO)CCCC1 C1(C(=O)NC2(CNC(C(C)OCC3CC3)=O)CCCCC2)CCC(C)(F)CC1 C1(C2CCCN(C(=O)C(c3ccccc3)=O)C2)(NC(C(C(C)C)O)=O)CC1 c1(C(CC(=O)NCC2(OC)CN(C(C3CCCC3(F)F)=O)C2)C)c(C)noc1C c1(CN(C)CC2(OCC)CCOC2)cc(C(F)(F)F)cc([N+](=O)[O-])c1 N1(C(C(C=CC)O)=O)CCN(C(c2[nH]c(C)c(C(=O)OC)c2C)=O)C2CCCC12 N1(C(C2C(CC)C2)=O)CC(NC(C2CC(=O)N(CC3CC3)C2)=O)C(C)C1 CC(C)(CCC#N)C(=O)N1CCCCC(NC(c2cnc(Cl)[nH]2)=O)C1 c1(NC(CC2CCN(Cc3c(C)nc[nH]3)C2)=O)ccc(CCN(C)C)cc1 C12(CNC(=O)CCCCC3CC3)CCC(NC(=O)C=Cc3ccccc3)(CO1)C2 C12(NC(c3c(CC)occ3)=O)CCN(C(c3cc(C)ncc3C)=O)CC1C2 C(=O)(CC(=O)N(CCCOC)C)NCCO.C12(CC1)C(=O)NC2.C1(C)CC1 C(=O)(CCC1=NNC(=O)CC1)NCC(CC(C)C)(C)NC(=O)CC1CSCCS1 c1(C(C)(C)C)ccc(C(N2CCCC2CNC(C23CCC2C3)=O)=O)s1 C1(NCC2(O)CCN(C)C2)Cc2n[nH]cc2C(C(F)(F)F)C1 N1(C(CN(CC)CC)=O)CC2COCCC2(NC(=O)CC(C)(C)C#N)C1 N1(C(c2ccc(CS(C)=O)cc2)=O)CCCCC(NC(=O)C(N)=S)C1 CCC(C)C(C)C(=O)N1CCN(C(c2ccn(C3CCC3)n2)=O)CC1CCOC C1(CNC(CNC(=O)OC)=O)CCC(C)CN1C(C1CC2C=CC1CC2)=O CC(F)CC(=O)N1CCC(CNC(C2(c3cccnc3)CC2)=O)C1 CC1(C)CC(NC(c2ccc(-n3cnnn3)cn2)=O)CN1C(C1CC2(CC2)C1)=O C=CCCC(C(=O)NCc1cc(C)c(C)o1)NC(c1cnncc1O)=O C(CCCC(=O)N1CCCCC1CN(C)C(c1occc1F)=O)SC CCC(C)CCC(=O)N1CCC(C(N2CC(O)CC(O)C2)=O)(CF)C1 c1(C(=O)NC2CC(C(N3CC(C)C(O)CC3)=O)C2)c(F)cc(Cl)cc1Cl C1(NC(c2c(C)cc(C(F)F)o2)=O)CN(C(c2ccc[nH]2)=O)CC1N=[N+]=[N-] c1(C(=O)NC2C(C)CN(C(c3ncc(Br)cn3)=O)C2)cc2c(ncn2C)[nH]1 C(=O)(C(O)(C(C)C)C(F)(F)F)N(CCCNC(c1cc2oc(C)c(C)c2[nH]1)=O)C C(C(=O)NC1CC(=O)N(C)C1=O)(C(C)(C)C)NC(c1c(NC)cccc1)=O c1(CNC(c2ccnc(-c3cnn(CCF)c3)c2)=O)cncc(Br)c1 N1(C(c2n(C)ccn2)=O)CC(C2CCCCN(C(C3(C)CC4CC4C3)=O)C2)C1 C12(C(N(C3CCC(NC(c4n(CC)ncn4)=O)CC3)C)=O)CCOC1CCOC2 c1(C(=O)NOC2CCOC2)cc(Cc2ccccc2)n[nH]1 C(N=c1[nH]ccc(C#N)c1[N+](=O)[O-])C1(O)CN(C(C2(OC)CCC2)=O)C1 O=C(O)CCCCC(=O)N1CC(Cc2cccc(OC(F)F)c2)C1 c1(CCC(=O)NC2C(NC(C(=C(C)C3CC3)F)=O)C2)ccc(O)cc1 C(CCCCC(=O)NC1CC1)NC(CCCCOCCCNC(C)=O)=O CN1CCOC2(CN(C(c3n[nH]cc3CNC(C3CC=CCO3)=O)=O)C2)C1 O=C(C1=NOC(CNC(C2CSCC(=O)N2)=O)C1)Nc1ccc(Cl)c(O)c1 Cc1cnc(CNC(C2CN(Cc3ccn(-c4ccccc4)n3)CCO2)=O)cn1 c1(N2CCC(C(C)C)C2)nnc(-c2cnn(C)c2)n1CC1CCCCO1 N1(C(Cc2nc(C)[nH]n2)=O)CCN(C(c2cccc(CN(C)C)c2)=O)CC2(CC2)C1 C1(C(N(CCC)CCC)=O)CC2CC1CN(C(C1(CO)CCOC1)=O)C2 C1(CNC(c2nc(C)n(C)n2)c2nnnn2C)CC2CCC(C1)C2 Cc1ccccc1C(=O)NCC1(C)CCN(CCCC(C)(C)C)C1 CON1CC(C(=O)NCC2CC2NC(=O)Cc2ccc(OC(F)F)cc2)CC1=O N#Cc1cc(C(N2CCC(O)(CCNC(C3CC(F)(CO)C3)=O)C2)=O)cc(O)c1 N1(C(C(=O)N(C)C)=O)CCCC(C)(C(N2CC(O)C(F)C2)=O)C1 C(=O)(C1CCc2nccn21)N(C(CNC(=O)CCCC(F)(F)CO)C1CC1)C N1(C(C2CN(C(=O)NC)C2)=O)CC=CC(NC(c2cnc(CC(C)(C)C)o2)=O)C1 C1(NC(C(CC)O)=O)(CNC(=O)C(c2ccc(C)cn2)(F)F)CC2CCC1CC2 C1(C(N(CCCC)C)=O)CNC(=O)CN1C(C1CC1CC(C)C)=O c1(CCC(=O)NCC(CO)NC(c2c(CC)nc(C)[nH]2)=O)c(C)nc(O)nc1O c1(C(C(N2CCCCC2Cc2cn(C3CC3)nn2)=O)O)ccc(F)c(Br)c1 N1(C(CSCC=C)=O)CC=C(C(=O)NCCC2CCC(C)(C)C2)C1 c1(OC)c(C(=O)NC2COCC2NC(c2ccsc2CO)=O)cccc1C(F)F n1(CC)c(C(N2CCCC(CN(C)C(c3csc(C(C)=O)c3)=O)C2)=O)cnc1O c1(C(N2C3CCN(C(C(CC)C)=O)CC3C2)=O)ccc2c(c1)COCC2 C1(NC(CC(C)F)=O)CCCC(C(=O)NCC2(O)CCC2)C1 C1(CC)CC2(CCN2C(C2CCN2C(C2(OC(C)C)CCC2)=O)=O)C1 C12(NC(=O)Cc3cnccc3Cl)CCN(C(=O)C(=O)Nc3ncc[nH]3)CC1C2 N1(CC2C(=O)N2)CCNC(=O)C1(C)C.C1(N(C)C(C(C)(C)C)=O)CCCCC1 c1(C(=O)NC2(CNC(CC3COCC(C)O3)=O)CCC2)ccnc(Cl)c1N Cc1nn2cc(CC(=O)OCC(N3CCC(N=[N+]=[N-])C3=O)=O)nc2s1 c1(C(=O)NC(CNC(C(C)N(C(C)=O)C)=O)CO)ccnn1C(C)C c1(CC)cc(C(=O)NCCCCC(C)NC(=O)Cc2ccnn2C2CC2)ccc1F CC(CCCO)NC(=O)CC1CC(NC(=O)CCn2cnnn2)C1 c1(CC)nocc1C(=O)NC(C1CC(C(=O)NCC(C)(C)CO)C1)C C1(NC(C(C)Cc2ccccn2)=O)CCN(C(C23CC(F)(C2)C3)=O)CC12CCC2 CC(CC(=O)N1CCC1CNC(=O)Cc1ccc2occc2c1)C(F)(F)F c1(C(=O)NC(C)CNC(c2cc(C3CC3)ns2)=O)cccc(S(N)(=O)=O)c1 CC(C)C(C#N)C(=O)NC1(COCCC(=O)NOC2CCC2)CCCCC1 C1(CNC(C=CCCC)=O)CC(C)N(C(c2cccc(OC)n2)=O)C1 c1(CC(=O)NC(C)CNC(C2(n3ncc(Br)n3)CC2)=O)c(C2CC2)cnn1C c1(CC)nnc(C(=O)NC(C)(C)CCNC(c2cn(CC)cn2)=O)s1 N1(S(C)(=O)=O)CC2CN(C(=O)CN3CCC(Nc4ccccc4S)C3)CC2C1 CCC(CNC(=O)CC1CCC(=O)O1)(CC)NC(C1CCCC1O)=O N1(C(c2cc(OC)n[nH]2)=O)CC2(CCC(CNC(=O)CC(F)(F)F)O2)C1 c1(C(N(CC(CC)NC(=O)CCN(C)C(C)=O)C)=O)ncn2c1CCC2 CN1CC2CCCC(C1)N2C(C1(C)CCCN1C(C1CCOC1)=O)=O c1(C(=O)NCCCCNC(C(c2cn(C)nc2)O)=O)ccc2c(c1)OCC2 C1(C(=O)NC(c2cnsc2)C)(CC)CCN(C(=O)CC2CC3(CC3)CO2)CC1 C1(C(N2CCC(OC)CC2)=O)C(C2CC2)CCN1C(c1nc(O)sc1C)=O C1(NC(c2c(OC)ccs2)=O)CCCC(NC(c2ccc(C3CCC3)cc2)=O)C1 N1(C(C2CN(C)C(=O)C2)=O)CCN(C(c2ccn(C(C)(C)C)c2)=O)CC1CCO c1(N(CCCCCCC)C)ccc(S(=O)(=O)N2CCC(C)C(CO)C2)c(Cl)c1 N1(C(CCC=C)=O)CCC2CCCC(C1)N2C(=O)C(C)Oc1ccc(Cl)c(Cl)c1 CC(C)(C)C(=O)N1CCCC1CN(C1CC1)Cc1ncc(C(=O)O)o1 c1(CC)nc(=N)[nH]cc1C(=O)NC(C)CC(C)NC(c1cc(Cl)c(Cl)n1C)=O C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCC(C)(NC(c2cnn(CCC)c2Cl)=O)C1 N1(C(C2C(=C)C2)=O)CC(NC(=O)C=Cc2cnc(C)s2)C(n2ccnn2)C1 c1(CN(CC(C)O)C(C2(NC)CCOC2)=O)ccc(F)cc1F C(=O)(CCCC(=O)N(CCN(C(=O)CC1CCCC(C)C1)CC)CC)OCC N1(C(C2CCCOC2)=O)CCN(C(c2cc(Cl)cc(Cl)c2)=O)C(CO)C1 C1(CCC(=O)NCC(C)(C)OC)CCN(C(=O)C=Cc2ccsc2)CC1 C1(NC(C(CC(=C)Cl)NC(=O)C(C)COC)=O)CN(C)CCN(C)C1 C=CCC(C(=O)N1CC(CC(C)(C)CN(c2cc(Cl)cs2)C)C1)c1ccccc1 N1(C(C(C)n2ccnc2)=O)CCC(N(C)C(c2csc(Cl)c2)=O)C2(CC2)C1 Nc1ccc(Cl)cc1C(N1CCCN(C(C23CCCC2(C(=O)OC)C3)=O)CC1)=O n1(CC(=O)OC)c(C)cc(C(=O)NC2CCN(C(=O)C3=CCCCC3)CC2F)c1C c1(C(NO)=O)c([N+](=O)[O-])cnn1CC(F)F.c1(OC)cccc(OC)c1Br N1(C(C2CCCO2)=O)CCN(C(=O)C=Cc2cccnc2)C(C2CCCC2)C1 N1(C(c2c(OC)c(Cl)ccc2)=O)CCC(C)(C)C(NC(c2occc2C)=O)C1 Cc1cc(=NC(=O)CC2CC3(C2)CN(C(c2ccc(C4CC4)cc2)=O)C3)[nH]n1C N#Cc1cccc(C(=O)NCCCN2CCC(O)C2)n1 O=C(CCCCCn1cc(-c2cnsc2)nn1)NC(C1(CO)CCCO1)=O N1(C(CC=CC=C)=O)CCN(C(c2c(Cl)sc(C)c2C)=O)CC1CC c1(NC(=O)NC2C3CN(CC)CC2CC3)ccc([N+](=O)[O-])cc1C(N)=O CC1(C)CC(C(N2CCC(NC(c3cc(Cl)cs3)=O)C(O)C2)=O)C(C)(C)O1 C12(NC(c3cncc(N(C)C)c3)=O)CCC(CN(C(c3cccc[n+]3[O-])=O)C1)C2 N1(C(c2n(CCC)ccc2)=O)CCOC(CCCNC(=O)Cc2cccs2)C1 Cc1cc(C(=O)NC(C)CCCNC(c2[nH]nnc2C)=O)c2ncccc2c1 C(=O)(C(O)CC(C)(C)C)NC1CCC(N(C)C(c2ccc(C(N)=O)cn2)=O)CC1 C1(NC(CNC(Cc2c(C#C)cccc2)=O)=O)CCC(=O)N(C)C1=O CCC(CC)CCCC(=O)N1CC2(CC2)CC1CNC(c1nc(C)nn1C)=O N1(C(CC(C(C)OC)NC(=O)CC2CC2)=O)Cc2ccc(C)nc2C1 Cc1ncc(C(=O)NC2CC(C)N(C(=O)CC3CCC(F)(F)C3)C2)c(C2CC2)n1 c1(OC)ccc(CN2CCC(C)(C(=O)NC(c3cncnc3)C)C2)c(C)c1OC N1(C(CC(=O)NC)=O)CC23CCCC2(C1)CN(C(=O)C(C)c1ccsc1)C3 c1(C(N2C(CNC(C(C)CC3CC3)=O)CC(F)(F)C2)=O)nnc2n1CCCCC2 N1(C(C2(C)COC2)=O)CCc2nn(C)c(C(=O)Nc3cccc4c3CCC4)c2C1 N1(C(c2cnc[nH]2)=O)CCS(=O)(=O)C(CCNC(C2CC(N3CC(O)C3)C2)=O)C1 C1(C(=O)NCC2N(C(c3c(CC)cno3)=O)CC(O)C2)CC2(CCC2=O)C1 C1(CN(C(c2cnncc2O)=O)CC)CCCN(C(=O)CCc2cnc(O)[nH]2)C1 CP(C)(=O)C1CCCCC1C(=O)NCC1CCN1C(=O)CC1(C2CC2)CC1 C1(NC(c2ccncc2Cl)c2n(C(C)C)nnn2)CCCCCCCCC1 N1(CC)CC(CNC(=O)CC2(C)CN(C(=O)CCN3CCCC3)C2)CC1=O C1(CC(=O)NOCCCO)CCCN(C(c2ncccc2Cl)=O)C1 C1(NC(C(CC)SC)=O)CN(C(c2ccc3nc[nH]c3c2)=O)C2(CCCC2)C1 c1(CNC(C(=O)Nc2ccc(-c3c(C)ncs3)cc2)=O)cc(F)c(F)cc1F c1(C(=O)NCC(CN(C(C(CSC)O)=O)C)C)c2c(nn1C)CCS(=O)(=O)C2 c1(NC(C)=O)c(F)ccc(-c2cccc(NC(C3CC(=O)N(C)C3)=O)n2)c1F C1(NC(C23CC(NC(Cc4nc(C)sc4)=O)(C2)C3)=O)CCOCC1C c1(OCC)ccccc1OC(C)C(C)OC.C12CCC(CC1)NC(=O)N2 C1(COC(c2c(=N)[nH]n(C)c2)=O)C[Si]2(CCCC2)CN1C(=O)OC(C)(C)C c1(C(N2CC(NC(Cc3n(C)cnc3)=O)C2)=O)ccnc(NC2CCC2)c1 C1(CCNC(C2CC2c2ccccc2)=O)CCN(C(c2ccncn2)=O)C1 C1(CNC(CC(CCC)O)=O)CN(C(c2ncn(C)c2C)=O)CC(C)(C)O1 C(=O)(CC(O)CC(C)(C)C)OC.c12nsc(n1)NC(=O)C2n1cc(Br)cn1 CC1CCC(CNC(=O)C(c2ccco2)NC(C2CCC2)=O)N1C Cn1cc(C2OCCC2C(=O)N(CCNC(=O)Cc2nnc(O)s2)C2CC2)cn1 CCCC(C(=O)N1CCCC1CNC(=O)C(c1ccccc1O)OC)NC(N)=O c1(C(=O)NCCOCCN(C(c2c(C)noc2C)=O)C)cc2nccn2c(O)n1 CCCC(O)CC(=O)NC1(CCNC(=O)COCc2ccnn2C)CCC1 c1(CCOC(C(C2CCCOC2)OCC)=O)cccnc1C N1(C(=O)NCC(=O)NC(C(=O)OCC)C2CC2)CCCC1CCOc1ncc[nH]1 CCCC(C(C(=O)NCC1CCOC1)N1CCCCC1CCP(C)(C)=O)OC C1(NC(c2ncc(C)cc2Br)=O)CCN(C(C2CCC(=O)O2)=O)CC12CCC2 C(=O)(C1=CC2CCCCCCC12)N1CC(C)C(CNC(=O)C=CCO)CC1 c1(C(=O)NCC(CC=C)NC(=O)CC(C)(O)C2CC2)c(C(F)(F)F)oc(C)c1C N1(C(c2n(C)cc(Cl)c2)=O)CC2CC1CN2C(C1CCOC(C)(C)C1)=O C#Cc1ccc(Cl)c(C(=O)NCC2CN(C(=O)C(CO)N(C)C)CC2C)c1 CCC(C)CCC(=O)NCC1CN(C(=O)Cc2cnc[nH]2)CC1C(F)(F)F c1(CC(=O)NC2C(NC(CCC=C(C)C)=O)C2)c[nH]c2ccc(F)cc12 C1(CCCC)CCCN(C(C2CC3CC3N2C(=O)Cc2[nH]cnc2C)=O)C1 c1(N2C(C(=O)NC(CC(C)(F)F)=O)CCC2)nc2ccccc2o1 c1(C(=O)NC2CC(C(F)C(=O)NCC3CCC(C4CC4)O3)C2)cc2n(n1)CCC2 c1(C(=O)NC2(C)CCCN(C(C3CCC4CC34)=O)C2)cn2cccnc2n1 C1(C(N2CC(F)(CNC(C3=C(C)CCCC3)=O)C2)=O)CC(C)c2nc(C)cn2C1 c1(NC(=O)NC(c2n(CC(C)C)ncc2)C)ccccc1COC(C)(C)C Cc1nc2cc(C(=O)NC3COCC3NC(c3cncc(N)c3)=O)c(F)cc2[nH]1 CN1Cc2ccc(C(=O)NCC3CCN(C(=O)CC4(O)CCOC4)C3)cc2C1 Cc1nc(-c2c(C)noc2C)sc1C(N1CC(CCNC(=O)C(O)C2CC2)C1)=O C1(NC(c2cc[nH]n2)=O)CC2(CCCCN2C(=O)CCc2ccc(F)cc2)C1 c1(C(=O)NCC(CC)NC(C2CC(C(C)(C)C)=NO2)=O)cc(OC)c(O)cc1C c1(NC2(CNC(c3cnc(C(C)O)s3)=O)CC2)ncc(Br)c(O)n1 C1(CCNC(C2ON=C(C)C2)=O)CCCN(C(c2cccn2C(C)C)=O)C1 C(=O)(C1=CC2(CCOCC2)C1)NC1C(O)CCN(C(CC(CCCCC)C)=O)C1 N1(C(c2cc(C)sn2)=O)CCC2CC2(C(=O)NOCCCOCCO)CC1 c1(C(N2CCC3(C(NC(C(CC)N(C)C)=O)C3)C2)=O)cc(C)cc2c[nH]nc12 c1(OC)ccnc(C(=O)NC2(CNC(c3cscc3C(N)=O)=O)CC2)c1F Cc1cnn(CC(C)NC(=O)NC(c2cn(C)nn2)c2cccs2)c1 C1(SCC(=O)NC2CCN(C(C3(C4CCCCO4)CCC3)=O)C2)CCOC1=O c1(OCC)ccccc1C1(CNC(=O)NCC(n2ccnn2)C)CC1 CC1CC2(CCN(C(=O)C(C)n3ccnn3)CC2)CN1C(=O)C=CC(=O)N(C)C C1(C(=O)NC(C)CC(=O)NC2(CCO)CCCCC2)CCOCC1(C)C Cc1ncc(CC(=O)N(CCCNC(C2C=CCC2)=O)C(C)C)[nH]1 c1(CNCC(C)=CC(=O)N(C(=O)C(N)=O)C)cc[nH]c1CCC C(N=c1ccc(S(=O)(=O)NC(C)Cc2ccccc2)c[nH]1)c1ccc(OC)cc1 CC1CN(C(=O)C(O)CC2CN(C(=O)C=CCN3CCCC3)C2)CC1(C)CO c1(C(N(C)CC2N(C(C3C(C)SCCC3)=O)CCC2)=O)ccc2c(c1)NC(=O)C2 C1(O)(CNC(CC(C)SC)=O)CC2CCC1O2.c12occc1C(=O)NC2 C(C(C(=O)NCc1ncco1)C(C)C)NC(C(CC=C)C)=O N1(C(CC(c2ccc(C(C)C)cc2)C)=O)CCC(C2CCS(=O)(=O)CC2)CC1 CON(CCC(=O)N1CCC(CC(N)=O)CC1)C(=O)CN1CCOCC1 Cc1cccc(C(N2C(C(=O)N=c3ccn(CCF)[nH]3)CC2C)=O)c1C#N c1(CC)onc(C(=O)N(CCC(C(C)C)NC(=O)C(C(C)C)NC(C)=O)C)c1C N1(Cc2n(CC)ccn2)CC2CCC1CN(C(c1cc(Cl)ccc1F)=O)C2 N1(CC2(C)CC2(Cl)Cl)CCC(=O)N(CCC2CCCC2)C1=O Cc1nn2cccnc2c1C(=O)NCC(C)(CO)NC(C1CC(C)(O)C1)=O C1(CC)(NC(=O)C=CC(=O)N(C)C)CCCN(C(=O)CC(C)SC)C1 C1(CC(N2C(CNC(Cc3c(C)ncs3)=O)CCC2)=O)CCC(C)(C)C1 c1(C(N(C2CCN(C(c3csc(=N)o3)=O)CC2)CCCC)=O)cnn2c1OCC2 C1(C(=O)NC(CC)C(N)=O)CCN(C(c2ccc(O)nc2C)=O)C(C)(C)C1 C1(C2CCC2)(C(=O)NCC(CC)(CC)NC(=O)CC2(N(C)C)COC2)CC1(F)F c1(C(=O)NC2CN(C(C34CCC(CC3)CC4)=O)CC2(F)F)ccc(F)cc1Br N1(C(c2ccc(SCCC)cc2)=O)CC2(CCN(C(=O)CC3(O)CCOC3)C2)C1 CC(CC(=O)N1CC2(CCCN(C(c3ncncc3Cl)=O)C2)C1)CC(C)(C)C c1(OC)nc(C)ccc1C(N1CC(C(C)NC(c2ccc(C(C)=O)[nH]2)=O)C1)=O C(CC(CC)C(=O)NC(C)CN(C)C(c1cc(C2CCOCC2)no1)=O)=CC N1(C(c2cc(=NC)[nH]cc2)=O)CCN(C(C2CCC(O)CN2C)=O)CC(O)C1 c1(C(=O)OCC(CCCC)C)cnc(NC(C)=O)c(OC)c1 C1(N(C)C)CC(NC(=O)CCCNC(=O)C=Cc2ccncn2)C1(C)C C(N=c1ncnc2[nH][nH]cc1-2)C1N(C(c2cc(C)c(F)cc2)=O)CCC1 C(C)(N=c1[nH]c(N2CCn3nncc3C2)nc2c1CSC2)c1c(OC)nsc1OC C(C(=O)N(CCC(C)NC(c1ccccc1F)=O)C)(C(C)C)SC c1(C(N2CCC(NC(c3ccc(OC)o3)=O)C2)=O)nccc(Br)c1C c1(-c2nccc(N(C(=O)C(O)C(C)(C)C)CC)c2)ccc2c(c1)CN(C)C2=O C1(C(N2C(C)(C(C)C)CC2)=O)COCCN1C(=O)C=CC1(C)COC1 C#CCCCC(C)C(=O)N1CC2(CC(NC(C3C(C#N)C3(C)C)=O)C2)C1 c1(C(N2CCC(C(N3CCC(SC)C3)=O)(CO)C2)=O)cccn2cncc12 n1(C2(N(C)CC)CC2)ccc(-n2cc(C3COCC3O)nn2)n1 Cc1cn2nc(C(=O)NC3CC(C)(NC(C4CCCC(F)C4)=O)C3)cc(C)c2n1 C1(C(N2CCC(C(CNC(C3(C(C)C)CC3)=O)(C)O)CC2)=O)CCCC12CCC2 C1(CNC(CCC=C=C)=O)CCN(C(c2cccn2C)=O)CC1C1CC1 N1(C(C2N(N=O)CCC2)=O)CC2CCC(N=c3ccn4c(Br)cnc4[nH]3)CC2C1 C12(NC(C3Cc4ccc(F)cc4O3)=O)CC3CCC(C1C2)N3C(C1(F)CC1)=O n1(C(C)C(=O)N(CCCCN(C)C(c2cc[nH]n2)=O)C)cnc(C#N)n1 C12(NC(CCCC(=C)C)=O)CCCN(C(=O)C=Cc3ccc(SC)s3)CC1C2 C(=O)(C(CC)C(F)(F)F)NC1(CC=C)CCN(C(=O)C(C)=C2CCCC2)C1 C(C(C)(C(=O)NC(c1ccccn1)C)NC(c1cccc(F)c1)=O)SC Cc1cc(C(=O)NCC2CC2NC(=O)CNc2nccs2)nn1C(C)C1CC1 C#Cc1ccc(C(=O)NCC2(F)CN(C(c3cc(NCC)ncc3Cl)=O)C2)cc1 C1(CNC(c2cc(Br)n[nH]2)=O)C2CN(C(=O)C(F)C3CCC3)CC12 Cc1ccc(OC(F)F)cc1NC(=O)NC1CCCCC1(C)O O=C(C1=CCOCC1)NC1C2CC3C1C3C2C(=O)NC1CC1c1cccnc1 C(=O)(C(CCC(N)=O)NC(N)=O)N1CC(NC(C(C(=O)OC)C)=O)C1 C(=O)(N(OC)C(C)CC)C1CC(SCCNC(CCC#C)=O)C1 c1(CC(OC)OC)cn(CCCN(C(=O)COCC2CCC2)C)nn1 C(=O)(C(CC=C)CC(C)C)N1CCC(CNC(CCOCC#C)=O)(OC)C1 c1(NC2CC(NC(=O)OC(C)(C)C)C(O)C2)cc(F)cc(F)c1.c12cccc(c1)N2C N#CC1(c2ccccc2)CCN(C(c2csc(C(=O)NCC3CC3)n2)=O)CC1.O N#Cc1cc(F)c(C(=O)NCC2CCCCC2NC(=O)CCC2CCC2)c(F)c1 CCCC(CC)CC(=O)N1CCOC(CNC(=O)C=Cc2cccc(C#N)c2)C1 C1(NC(C(C)(C)OC(C)C)=O)CC2CC(NC(C3CCN(C)C3C)=O)CC12 C1CCC(F)(F)CC1.c1(N(CC=C)CCC)nnc(COC)n1Cc1ccccn1 C(C(C(=O)NCCC#N)N(C(C#N)C1CC1)C)(C1CCOC1)OCC c1(C(=O)NC2C(C(N3CCC(C#N)C3)=O)C2)cc(Cl)cc(Cl)c1Cl C(=O)(CCCC(=C)C)NCC1(C(N2CCN(CC=C)CC2)=O)CC1 CCCC(CCCS(C)(=O)=O)C(=O)NC1CC(NC(c2ccc(CO)o2)=O)C1 CCC(CC(C)C)C(=O)NC12CCC(CNC(C3CCCC(=O)N3)=O)(CC1)OC2 c1(C(=O)NCC2C(OCC)CN(C(C3C(C)C3C)=O)C2)c(Cl)ccc(C)c1O N1(C(CC(C)(C)C#N)=O)CCC(C2CC(NC(C3(C)CC4(CCC4)C3)=O)C2)C1 c1(CNSC)cccc2c1OCO2.N12CCCC1C=CC=CC2.C1CC1 N1(C(c2ccc(C)s2)=O)CC2CC(NC(=O)Cc3cccc(C)c3Cl)C1C2 C(=O)(C(C)(C)CS(C)(=O)=O)NC12CC(CNC(C=NOC)=O)(C1)C2 Cc1cc(C(=O)N(CCCCN(C)C(c2nccnc2N)=O)C)c(C)c(C)c1 CC(C)CC(C)(C)C(=O)NCC1CN(C(c2cnc3ccoc3c2)=O)CCCO1 C1(COC)CN(C(c2ncoc2C)=O)CCC1NC(=O)CCNC(=O)OC N1(C(CCCOCC=C)=O)CC(C)CN(C(c2sccc2OC)=O)C(C)C1 C(=O)(C(F)(F)CCn1cccn1)NCC1C2CN(C(C(CCC)OC)=O)CC21 N1(C(C(CC=C)NC(c2cnc(CC)o2)=O)=O)CCC(CO)C(C)C1 N1(C(c2ncn(CC)c2)=O)CC2CC1CN(C(C1CC3CC1CO3)=O)C2 c1(NCC(C2CCCCC2)NC(C2CC23CCC3)=O)ncnc2ccc(O)cc12 C1(C(=O)NCc2ccc(C(=O)NC(CCC=C)C3CC3)o2)CC=C(C)CC1 N1(CC(=O)NCc2ncoc2C2CN(C(=O)C(F)C3CCC3)C2)CCC(O)CC1 CN1N=C(C(=O)NC2CCCCC2CNC(c2cc(Cl)n(C)n2)=O)CCC1=O c1(OC)cc(OC)cc(C(=O)N(CC(O)CNC(=O)CC(O)C(C)C)C)c1 S(=O)(=O)(c1c[nH]c(C(=O)O)c1)N1C(CC)CN(C(=O)COC(C)=O)CC1 c1(NC(=O)CC2CN(Cc3ccc(Br)o3)C2)cc(F)ccc1[N+](=O)[O-] C1(CCNC(=O)C(O)c2ccco2)CCCN(C(=O)Cc2ccoc2)C1 CC1(C2CCC2)CN(C(C2(C)CCCN2C(=O)COc2ccccc2)=O)C1 C(=O)(C1=CCOCC1)NC(C1(CNC(c2cncn2C)=O)CC1)C O=C(C1=CCCS1)NCc1cccc(CNC(C2CCCS2(=O)=O)=O)c1 N1(C(C(Cc2c(C)n[nH]c2C)C)=O)CCC(NC(=O)C=CCO)C(C)(C)C1 C(=O)(CS(=O)(=O)N1CCCCC1)NCC(C1CCC1)NC(C(C)=C1CCCC1)=O N1(C(C(CCC)CC)=O)CCC2C(CCN2C(c2ccc(C)c(C)n2)=O)C1 c1(C(=O)NCCC2(CNC(C(=O)C=Cc3cccs3)=O)CC2)cc2n(n1)CCO2 C(=O)(CC(F)(F)C(F)(F)F)N(CCCNC(c1oc(C(=O)OC)cc1C)=O)CC C1(C(N2CC(N(C(c3c(C)ncnc3)=O)C)C2)=O)CCOC2(CCCCC2)C1 Cc1c[nH]c(C(=O)NCCC2CN(C(C3C(C)CC3C)=O)C2)c1 Cc1cc([N+](=O)[O-])c(NC(=O)CCN2CCCC(C(N)=O)C2)cc1C#N c1(NC(CCCOC)C)cc(NCC(C)C(F)(F)F)ncn1 N1(C(c2n(CC)nc(C)c2)=O)CC2CCC2(CNC(c2cc(C3CC3)ns2)=O)C1 C1(C(=O)NCC2(O)CCN(C(C3(O)CCC(CC)C3)=O)C2)CN2CCN1CC2C C=CCC(CNC(C1(OC)CCC(C)C1)=O)C(=O)NC1CCC(N(C)C)C1 C1(C(=O)NC2(C)CN(C(C3(n4cccn4)CCCC3)=O)C2)COC2(CO)CC1C2 C1(C(=O)NC(c2ncnn2C)CC)CC2(CCC2)CN1C(c1n[nH]c(C)c1C)=O c1(C(C)(C)C)ccccc1C(=O)NC1CCCCC1NC(C1CCOC(=O)N1)=O N1(C(CNC(N)=O)=O)CCN(Cc2cc(Br)c[nH]2)C2CC12 CCCC(C)CC(=O)N1CC(C)(C)CC1CC(=O)N(CC(O)(CC)CC)C c1(CC(N2CCC(C(C)NC(CC=C(C)C)=O)C2)=O)cccnc1C(F)(F)F C1(O)(CN(C(c2ccc(C(OC)OC)o2)=O)C)CCCN(C(=O)C(O)C(F)F)C1 C1(CC(N)=O)CN(C(C2C=CCN2C(C2C3COCC23)=O)=O)CCO1 C(C(=O)NC(C1CC(NC(C2CC=CC2)=O)C1)C)(C(C)(C)C)SC N1(C(C2(CC#C)CC=CCC2)=O)CCCN(C(=O)C(O)COC)CC1 C1(CC)C(=O)NCCN1c1ccc(CNS(=O)(=O)CCCN2CCOCC2)cc1 c1(C(=O)NCC2CCCCN2C(=O)CCCc2cccnc2)cc(Cl)nc(Cl)c1 C1(OC)CN(C(=O)CCCn2cncn2)CC1NC(=O)Cc1ccn(C2CC2)n1 c1(OCCC)ccc(CNC(=O)C(c2ncsc2Br)N2CCC2(C)CC)cc1 C(c1cccc2c(OC(F)F)cccc12)=CC(=O)Nc1c(N)ccc(Cl)c1Br C1(NC(c2cc(COC)cn2C)=O)CN(C(c2ccc(F)c(C)c2)=O)CCC1F N(S(=O)(=O)N(C)C)CC(=O)NCCCN(C)C(c1cc(Cl)ns1)=O C1(C(CNC(C(COC)OC)=O)(C)C)CCCCN1C(c1cc(OC)ccn1)=O N1(C(Cn2c(C)ccn2)=O)CCC(C)C(CNC(c2ccc(C3CC3)o2)=O)C1 CC1CN(C(c2cc(O)cc(O)c2)=O)CCC1NC(=O)CCc1cnc[nH]1 CC1CCCC=C1C(=O)NC1CCN(C(=O)CCc2nc[nH]n2)CC1CO c1(OCC)ccc(-c2ocnc2C(=O)NCCC2CCCN(C)C2)cc1 c1(C(=O)NC2CN(C(C3C(C(=O)OC)CC3)=O)CC2O)cc2nc(F)ccc2o1 C=CCC(CC)C(=O)NCC1(F)CCCN(C(c2ccc(C3CC3)nc2)=O)C1 c1(C(=O)NCC(CNC(COC(CC)C)=O)C)cn(C)c2ccc(F)cc12 C1(CC)(CC)CC(C(N2CCCC2C(C)NC(=O)Cc2cnnn2C)=O)C1 Cc1ccc(Cl)c(C(N2CCCC(NC(=O)CCC3CCC(=O)NC3)C2)=O)c1 c1(CNC(c2nc(C(=O)OC)sc2)=O)cccc(C)c1F CCCC(CC)CC(=O)NC1CN(C(=O)Cc2ccnn2C)CC1(C)C c1(C(N2CCC(C(C)Nc3nccc(OC)n3)C2)=O)c(Cl)oc2ccccc12 C1(NC(C(CCC)OC)=O)CCCN1NC(=O)C1(OC)CCCSC1 c1(C(=O)NCc2ccccc2CNC(C2CC=CCO2)=O)cnc2[nH]ncc2c1 O(N1CCC(NC(=O)C(C(C)C)NC(C2CCCC(CF)C2)=O)CC1)CC C(C(C)C(F)C(=O)N1CC2C(C)C2C1)NC(CN1C(C)CCC1)=O C(C(=O)N(CCC(=O)NC1CCN2CCCCC12)OC)c1cn(CC)nc1 C(=O)(C(C)C(O)C(C)C)NCC(CNC(c1cn(C(C)C)nn1)=O)OC CC(C)C(C(=O)NCC1CCC(N(C(=O)CCC2CC2)C)CC1)C1CCC1 C1(NC(C2N(C)C(=O)CC2)=O)CN(C(c2cc(F)c[nH]2)=O)CC12CCC2 N1(C(=O)CCNCC2(O)CNC2)CC(c2ccccc2)CC1=O O=C(C1=C(Cl)CC1)NC1CCCC1CNC(c1cnn[nH]1)=O N1(C(c2cc(CC)oc2C)=O)CC2(CCC(NC(c3cc(C)ncn3)=O)CC2)C1 C12(C(=O)NCC(Cn3cc(-c4ccc(F)c(Cl)c4)nn3)OC)CC(C)(CCO1)C2 C(c1ccc(C(N)=O)o1)=CC(=O)NC(CNC(C(C)NC(=O)NC)=O)(C)CO C#Cc1ccc(C(N2CCN(C(c3cc(C(F)(F)F)n(C)n3)=O)C(C)C2)=O)cc1 CC(CC(F)F)C(=O)NCCN(C1CCCC1)C(c1c(Br)nnn1C)=O c1(NC(=O)Cc2ccc(Br)nc2)cncc(CNC(=O)NC2C(C#N)CC2)c1 C1(NC(C(C2CC2)OCC)=O)CC2CCC1N2C(c1ccc(C)c(C(C)=O)c1)=O c1(C(N2CCCCC2c2cccs2)C(=O)NCCC)ccc(F)cc1Cl c1(C(N(CCCNC(C2(CC)COC2)=O)C)=O)cccc2c1CCOC2 c1(C(=O)NCC2CCN(C(c3nccc(C)c3)=O)C2)c(F)ccnc1F Cc1cnc(C#N)c(NC(C2CC23CN(Cc2ccnc(Br)c2)C3)=O)c1 C1(C(N2CCC(C(=O)NC)C2)=O)CCCN(C(c2cccc(C(=O)O)c2)=O)C1 C1(NC(C(C(C)O)C)=O)CN(C(C2CC(F)(F)C2)=O)CCC12CCC2 C(C#CC1CC1)NC(C1C(C(C)NC(=O)OC(C)(C)C)C1)=O c1(C(C)=O)ccc(C(=O)NC2CC(NC(C3(S(C)(=O)=O)CC3)=O)C(O)C2)cc1C c1(C(=O)NCCN(C(C2(CC=C)CC2)=O)C2CC2)ccc(C#N)cc1C c1(OC)ccc(OC(C)C(N2CCC(CCNC(C34CSC(C3)C4)=O)C2)=O)cc1 N1(C(c2c(CNC(Cn3ncc(C)c3)=O)ocn2)=O)CCN(C)CC(C)C1 C12(C(=O)NC(C(C)(C)NC(CS(=O)(=O)NCC)=O)C)CCC(C(F)F)(CC1)CC2 c1(OC)ccc(Cl)c(C(N2CCN(c3ccncc3)CC2)C(=O)NCC2CC2)c1 N1(C(CSc2nc(C)[nH]n2)=O)CC(NC(c2ncccc2C(C)(C)C)=O)C(C)C1 c1(C(=O)NC2(CC=C)CCN(C(=O)C=Cc3cn[nH]c3)C2)cc(OC)cc(F)c1 N1(C(C(c2nccn2CC2CCN(C3CC3)C2)C)=O)CCC(C(N)=O)CC1 n1(CC(N2CCC(C)(c3onc(C)n3)CC2)=O)ccc2ccccc12 C(CC(C)C)(C(=O)N1CCC(C(=O)NCCCC(O)CO)C(O)C1)OC Cc1cc(C(=O)NC(C)(C)CC(=O)Nc2cccc(C)c2C)cnc1O c1(N(C)C)ccc(=NC(=O)N2CCC3(C)C(C2)C3(Cl)Cl)[nH]n1 C1(C(=O)NC(CNC(C=CCOC)=O)(C)CC(C)C)CCC12CCOCC2 C1(c2n(CC3C(C)C3)nnn2)(NCc2csnn2)CC2(CSC2)C1 c1(CC)ccc(C(=O)N(CCCNC(c2ccc(COC)nc2)=O)C)cc1N C1(CNC(c2ccc(COC)s2)=O)CCC(C)N(C(C2(C)CC3(CC3)C2)=O)C1 N1(C(c2cc(C(F)F)no2)C(=O)NCC)CCN(C)CC1CC c1(C(=O)NCC(C(=O)N(C2CCCC2)CCOC)C)cnncc1C c1(COC)sc(N2CCN(Cc3noc(-c4ccco4)n3)CC2)nc1C Cc1nc(=NC2(c3ccccc3)CCN(C(c3c(C)nc(O)nc3S)=O)C2)s[nH]1 N1(C(C(c2ccccc2)OC)=O)CCCC1(C)C(=O)Nc1ccsc1C(N)=O Cc1nc(N(C)Cc2cc(C)on2)cc(N2CCC(Cl)=C(Cl)C2)n1 N1(C(C2(CC)CCCN2C(=O)CC2CCOC2C)=O)CCCCCCC1C CCC(CC)CC(=O)NCC1CN(C(C2CC(C)(O)C2)=O)CCN1C c1(SC)ncc(CNC2CC(NC(c3cc(I)ccc3Br)=O)C2)c(Cl)n1 C1(C(=O)NCCCC=CC)CC(NC(=O)CCC(=O)N(C)C)C1(C)C N1(C(C2CNC(=O)O2)=O)CCC(F)(CNC(=O)C(F)(F)c2nccs2)CC1 c1(N(C)C)ncc(C(=O)NC2CCN(C(=O)Cc3ccc(O)cn3)CC2)cc1Cl c1(CSC)ccc(C(=O)N(C2CN(C(=O)C(C)CSc3cccnc3)C2)C)cc1 N1(C(C(c2ccc(O)cc2)=O)=O)CC2(CCC2NC(c2ccc([N+](=O)[O-])o2)=O)C1 c1(C(N2CC(CCNC(C(=O)NC(C)C)=O)OC(C)C2)=O)cc(F)cc(F)c1O c1(C(C)C(=O)NCCN(C(=O)C(F)=C2CCCC2)C2CC2)c(F)cccc1F c1(C(N(CCNC(C(C2CCC2)OC)=O)C(C)C)=O)cc(CS(C)(=O)=O)c(C)s1 N1(C(CSCCCC)=O)CCN(C(=O)C(CCC)NC(N)=O)CC(C)(C)C1 O=C(CCCC(F)(F)F)NC1CN(C(C2CC23CC(F)(F)C3)=O)CC1C(F)F c1(C(N(c2ccc(C)c(C)c2)CC(C)C)=O)cnc2n(c(=O)c1=O)CCCC2 c1(COC)ccc(C(C(=O)NC2CC2)N(C)CCN(C)C2CC2)o1 C(CNC(c1ccccc1F)=O)(CC(=O)NCCOc1cccnc1)OC N1(Cc2c(OC)ccc(Br)c2)CCOC2(C1)CN(c1ncc(C)cn1)C2 CC1(C)CN(C(C2CC3CC3C2)=O)CC1NC(=O)C(c1ccc(F)cc1)C1CC1 c1(OC)cccc(O)c1C(=O)NC1CCCCN(C(C2CSCCS2)=O)C1 C1(OC)CN(C(c2nn[nH]c2C(F)(F)F)=O)CC1NC(C1CCCCCC1)=O N1(C(c2cc(OC)nn2C)=O)CC(NC(c2c[nH]cc2C(C)(C)C)=O)CC(C)C1 C1(C(=O)NCc2cccc(C(=O)NCCC3CCC(C)C3)n2)CC(C2CC2)=NO1 C1(=O)CCC(Cc2ccccc2)O1.N1(C(=O)OC(C)(C)C)CCC(C)=C(Br)C1 Cc1noc(C(F)F)c1C(=O)NC1CCCC1CNC(C12CC(F)(C1)C2)=O c1(C(C)(C)C)cc(N2CCC(CCNC(C3(C)CC3(F)Cl)=O)C2)ncn1 CC1CN(C(=O)CCOCCN(C)C)C(C)CN1C(c1cc(O)nn1C)=O c1(SC)c(NC(=O)C(C)(C)C2CCN(C(c3coc(N(C)C)n3)=O)C2)cnn1C N1(C(COC)=O)CC(OC)C(C(=O)NC(c2ccns2)C)C1 Cc1nnc(CNC(=O)C(c2cn(C)nn2)NC(c2csnn2)=O)s1 c1(NC(c2c(C)cccc2)CCO)nc(=NCCC(C)F)[nH]c2c(C)nn(C)c12 C1(NC(COCCCCCC)=O)CC(NC(=O)COCC(C)(C)C)C(O)C1 C(=O)(CCC(C)(C)F)NCCC1CCN(C(C2CN(C)C(=O)C2)=O)CC1 C(=O)(C1COc2ccccc21)N(CCN(C)C(C1CCC(c2cc[nH]n2)O1)=O)C c1(NC(CC2OCCN(C(CCCC#C)=O)C2)=O)c(OC(F)(F)F)cccc1F Cc1ccc(C(C(=O)O)NC(c2c(C)n[nH]c2C)=O)cc1 C1(NC(c2c(CC(=O)OC)occ2)=O)CCN(C(=O)Cn2cncc2C)C(C)C1 CCC(C)CCCC(=O)NC(CCC1CC1)C(=O)NCC(C)(CC)CC Cc1cn2c(C(=O)N(C)CCOCCN(C(=O)CN(C)C)C)cnc2s1 c1(C(=O)NC(C)CN(C(=O)C=C(Cl)Cl)C)cc(C(C)(C)O)ccn1 CC(C)(F)CCC(=O)N1CCC(CNC(c2cc(Cl)ccc2Br)=O)CC1 C(=O)(C(F)C(C)CNC(=O)CCN(C)CCO)N1CCC(CCOC)CC1 c1(CC)scnc1C(=O)NC(CN(C(=O)COC1CC1)C)Cc1ccccc1 c1(OCC(N2CCC(NC(=O)C(F)=CCCF)CC2)=O)ccc(Cl)c(C(F)F)c1 CC(CN(C)C)CCC(=O)NCC(C)CC(=O)N1CCCC1(C)C C1(NC(c2c(C)cc(C)o2)=O)COC2(CCN(C(C3(C(N)=O)CCC3)=O)C2)C1 CC1=C(C(=O)NCC2CCCC2NC(=O)Cc2nonc2C)CCCO1 C1(NC(c2c(C)nc(CC)s2)=O)CN(C(c2nncs2)=O)C2(CCC2)C1 Cc1cc(C(=O)NC2(CNC(C3CC3F)=O)CC2)ncc1C(F)F C=CC1(C(N2CC(NC(c3cccc(F)c3SC)=O)CC(F)C2)=O)CCCCC1 S(=O)(=O)(c1[nH]c(=NC2CCCN(C3CCOCC3)C2)ccc1Br)NC1C(C)C1 C=C(C)C(C)(O)C(=O)NC(CNC(=O)Cc1ccc(Cl)cc1)C1CCC1 Cc1c(F)ccc(C(N2CC3CC3(C(=O)N=c3cnn(C)[nH]3)C2)=O)c1F N1(C(c2nc(CC)oc2)=O)CC2(CCN(C(C3CCN(C)C3)=O)CC2)CC1C c1(OC)cccc(C(CC(=O)O)Nc2ccnn2CC2CCC2)c1Cl N1(C(C(C)OCC2CC2)=O)CC(C(=O)Nc2cc(C#N)ccc2O)CCC1(C)C O=C1COC(CNC(C2CC(O)CN2C(c2ccc(S)cc2)=O)=O)CN1 N1(C(C(C)n2ccnc2)=O)CC(CNC(C2(C)CCN(C)CC2)=O)C(C)(C)C1 N1(C(C=C(C)c2ccco2)=O)CCCN(C(=O)C(C)(C)NS(C)(=O)=O)CCC1 N1(c2cc(N(C)CC3CCCS3)nc(C)n2)Cc2cccn2C(C)C1 c1(CC(N2CC(CCCOC)OCC2)=O)c(NC(C2CC2CF)=O)cccc1F c1(OC)ccc(OCCC(=O)NCC2(C(F)F)CCN(C(=O)C(C)CO)C2)cc1 Fc1cccc(C2CC(NC(C3CCCCCC3)(c3nnnn3C3CC3)C)C2)c1 N1(C(COCCCC)=O)CC2CCCC2(C(=O)NCCc2cnnn2C)C1 C1(C2(C(c3cc(-c4ccoc4)[nH]n3)=O)CC2)CCCCN1C(C1C(=O)NCC1)=O C1(NC(c2cnn(C(C)C)n2)=O)CCC(C(N2CC3C=CC3C2)=O)CC1 C1(CNC(c2cc(OC)n[nH]2)=O)CC(NC(=O)CCCOC)C12CCC2 c1(NC(C2(O)CCN(Cc3c(N(C)C)cccc3)C2)=O)cc(C)c(Cl)cc1F N1(C(C(CO)NC(c2c(C)c[nH]n2)=O)=O)CCN(C)C2(CCC2)C1 c1(C(N2CCC(NC(C3C(C)CCO3)=O)(CF)C2)=O)cnc2c(c1)NC(=O)CS2 c1(-c2c(C)cccc2)cc(=NC(=O)CC2(C)CN(c3ccc(I)cc3Br)C2)[nH][nH]1 c1(NC(=O)CC(C)(C)C)ccc(CC(C)C(=O)NC2CC2(C(=O)OC)CO)cc1 CC(C)C(F)C(=O)NCCC1CCCN(C(c2ccc(Cl)cc2)=O)C1 c1(C(N2CC(C(C)NC(=O)CCN3CCCCC3)C2)=O)csc2c(F)cccc12 Cc1nc(C(=O)NC2CC(NC(C3CC4CCC4C3)=O)C2)c2ccnc-2[nH]1 c1(CC)nn(C)c(Cl)c1C(=O)NC1CN(C(c2cnncc2C)=O)CCC1C N1(C(c2ccc(F)cc2F)C)CC=C(CCNC(C2C=CC=CC=C2)=O)CC1 CCCCCCCC(=O)NC1CC12CCN(C(=O)CC(=O)OCC)CC2 O=C(C1CCCc2ncccc21)NC1C=CCN(C(c2cccnc2O)=O)C1 c1(OC(C)C)ccccc1-c1cn(CCCNC(=O)CCc2cccn2C)nn1 C12(C(N3CCC(C(C)NC(CC4N(CC)CCC4)=O)CC3)=O)CCC(CC1)OC2 N1(C(C(COC)N(C)C)=O)CCC(O)(CNC(c2ccc(O)nn2)=O)C1 N1(C(C)C)CCCC1C(=O)NC(C)CNC(C1CC1c1cncn1C)=O C1(NC(CC(C(C)C)O)=O)CN(C(C2CCC(C)O2)=O)CC2(CC2)C1 c1(C(=O)NCC2(O)CCN(C(C3C(C)CC3)=O)CC2)csc(S(N)(=O)=O)c1 C(=O)(C(C)CS(C)(=O)=O)N(C(CN(C(c1c(C(C)C)ccc(Cl)c1)=O)C)C)C C=Cc1ccc2c(c1)CN(CC(c1cccc(C)c1)C)C2 C1(C)(NC(c2cc(C)ns2)=O)CCCCC1C(=O)NCc1cnccn1 C1(C(C)NC(=O)C(C2CCC2)Sc2cn[nH]c2)CCN(C(=O)COC(C)(C)C)C1 Cc1ccc(C(=O)NCC2CCCCN(C(=O)C(F)C(C)C)C2)c2cccnc12 S(=O)(=O)(c1cccc(=NCC2CCN(C3CC3)C2)[nH]1)NCC(c1cn(C)nc1)O C=C(C)CC(C(=O)N1CC(C)(C(N2CC(F)C2)=O)C1)OC c1(-c2cccc(C(=O)NCCCC#C)c2)ccc(F)c(CCO)c1 CC1C=C(C(=O)NC2CCC(NC(=O)CCP(C)(C)=O)CC2)CC1 c1(C(N2CC(OC)(CNC(=O)C(C)(O)C3CCOC3)C2)=O)ccnnc1C c1(C(=O)NCCC(C)NC(CC(C(F)(F)F)OC)=O)[nH]c2cc(C)ccc2c1C N(C(=NCCCF)N1CCC(c2ccccc2)(C(F)(F)F)C1)C1CC1.FCC c1(C(C(=O)NC(CC)C)N(c2ccc(Cl)o2)CCc2ccccc2)nncn1C N1(C(c2cc(CNC(CCCC)=O)oc2)=O)CCN2C(=O)CCC2C1 C1(C(=O)Nc2c(C)cc(Br)cc2)CCC2(CCOC2)O1 C1(N(C(Cc2n(C)ncc2)=O)C)CCC(NC(c2ccns2)=O)CC1 c1(-c2nc(C)sc2)ccc(S(=O)(=O)N2CCN(C(C)C)CC(C(=O)O)C2)cc1 C(=O)(C#CC1CCOC1)N1CCCC(CNC(C=Cc2cn(C)nc2)=O)C1 c1(NC(C2CC(n3cc(CCC(C)(C)O)nn3)C2)=O)nc2cccnc2s1 C1(C(N2CC(O)(COC)C2)=O)CC2(C1)CN(C(c1ccn(C3CC3)n1)=O)C2 c1(C(N2CC3C(NC(C4ON=C(CC)C4)=O)(C3)C2)=O)cnc2[nH]c(O)nc2c1 c1(CC)cnccc1C(=O)NC(C)C(C)NC(=O)C1=CCSC1 CCCCCCCCCCC(=O)NC(C)(C)CNC(C1COC2(C)CC1C2)=O c1(C(NOCC(=O)OCC)=O)coc2c1CN(C(C1CNC(=O)N1)=O)C2 N1(C(c2conc2C(F)(F)F)=O)CCC(C(=O)O)C(NC(=O)C(F)(F)F)C1 N1(C(C2(OC(C)C)CCC2)=O)CCC(C)(CC(=O)NCC2(O)CCC(C)C2)C1 c1(C(=O)NC(C(=O)NCC(C)(C)C2CCCC2)CC2CCC2)cc(F)ccc1O c1(C(N2CCC(NC(c3c(Cl)cnc(C)n3)=O)C(C)C2)=O)cnn2ccccc12 c1(C(=O)NC2CCN(C(c3cn4ccnc4s3)=O)CC2)cnc2ccc(F)cn12 C(=O)(C#CC1CCOC1)N(CCNC(C(C)Oc1ccc(F)c(F)c1)=O)C1CC1 C=C(C)CCCC(=O)N1CCCC1CN(C(=O)Cc1c(C)cnn1C)CC Cc1cc(=NCCC2COC(C)(C)C2)[nH]c(NCc2ccn(C(C)C)n2)n1 c1(C(=O)NCC(=O)NC2CC(CNC(C(CC)F)=O)C2)ccc(N)cc1 C1(C(=O)NCC(CCC)(C)O)C2CC(O)C(C2)N1C(c1c(C)cccc1F)=O c1(NCC)ccc(C)cc1C(=O)NC1CC1NC(=O)C(CCSCC)NC=O N1(C(COCC(=C)C)=O)CC(CC(=O)N(CCN2CC=CC2)CC)CC1C CC(C)CC(CNC(C1CC(=O)CN1C(c1cccnc1S)=O)=O)CO c1(OCC)cccc(CC(CC)N(c2n(C)c(COCC)nn2)C)c1.C1(C)(O)CC1 c1(C(=O)NC(c2cn(C)nn2)C(=O)NC(c2cccnc2O)C)ncc[nH]c1=O c1(OC(C)C(=O)NCC(=O)Oc2ccc(I)cc2)ccc(F)cc1Br C1(NC(C=C(CC)C)=O)CCSC12CN(C(=O)COCc1cccc(C)c1)C2 C(CCS(N)(=O)=O)c1cn(CCNC(=O)C(c2nnc(C)o2)C2CCCCO2)nn1 C1(NC(c2c(C)cco2)=O)CCCC(N(C)C(c2cccc(CF)c2)=O)C1 c1(C(=O)NC(C2CCCC2)CNC(CC(C(=C)C)OCC)=O)cnn2c1CCC2 CC1CCC(C)C1NC(=O)C(C)CNC(C1OCCC1C(C)C)=O S(=O)(=O)(CCC(F)(F)F)NC1(C(=O)Nc2cccc(N3CC(O)C3)c2)COC1 C1(C(=O)NCCC2N(C(c3cccc(CCC)c3)=O)CCC2)CC(=O)NC(C)C1 C1(F)(CNC(c2nc(C)sc2C)=O)CCN(C(=O)CNC2CCCCC2C)CC1 c1(C(N2C(CN(C(C3CC34CC4)=O)CC)CCCC2)=O)c[nH]c2cccc(C)c12 c1(C(=O)NC2(C(=O)NC(c3cc(C)on3)C)CC2C)cnc(O)c(F)c1 C(=O)(CS(=O)(=O)CCO)N1CCC(CNC(C2=C(C)OCC2)=O)(CO)C1 Cn1cncc1C(N1CCC(CCC(=O)Nc2cnnn2-c2ccccc2)C1)=O C(=O)(C(C)C(C)c1ccc(Cl)cc1)NCCCN(C(C1(OC)CC1)=O)C1CC1 C1(CC)C(NC(=O)CCOCC(C)C)CCCN1C(C1CCS1(=O)=O)=O CCC(CC)(C(=O)NCC1CCCC1NC(=O)C=CSC)c1ccc(Cl)cc1 c1(C2C(NC(C3CCCC3NC(C3C4COCC34)=O)=O)C2)ccc(Br)cc1 C1(C(=O)NCc2nc(CC)oc2)CC2CCC(C1)N2C(C1CS(=O)(=O)C1)=O C(=O)(C1=NOC(C)C1C)NC1C(NC(c2cccc(CC)n2)=O)COCC1 C1(NC(c2c(C#N)scc2)=O)CCCCCN(C(=O)C(O)CN2CCCC2)C1 C1(C(N(CCCNC(c2ccc(C3CC3)o2)=O)C(C)C)=O)CCOC(=O)N1 CC(C)(C)CC(CNCc1cn(Cc2ccccc2)nn1)CO c1(C(=O)Nc2cccc(NC(c3c(CC)nn[nH]3)=O)c2)ccc([N+](=O)[O-])[nH]1 C1(C)(CC)CN(C(=O)C(CC(C)C)NC(=O)CC2(O)CCOCC2)CCO1 C1(NC(CC(C=C)(C)O)=O)CCCC12CN(C(C1(C)CCS(=O)(=O)CC1)=O)C2 N1(C(C(C)c2cccs2)=O)C(CC(=O)NCC(C)C(C)(F)F)C2CCCC12 C1(CNC(CCSC)=O)C2CCC1CN(C(=O)CN1CCn3ccnc3C1)C2 C1(CCC)CN(C(C2(C(=O)OC)C=CCC2)=O)CCN1C(c1cnc[nH]c1=N)=O c1(C(C(=O)OC)NS(=O)(=O)C2CC2)ccc(NC2C(C)(C)C2(C)C)cc1 C1(CN(C(COC)=O)C)CCN(C(=O)CCCCc2ccc(OC)cc2)CC1 N1(C(Cc2cc(C)nn2C)=O)C2CCCC1CN(C(=O)CCCS(C)(=O)=O)CC2 Cc1oc(CNC(C2(F)CCCC2)=O)nc1C(=O)N(C)CCc1cnc[nH]1 C1(NC(c2ccn(C(C)C)n2)=O)C2CCN(C(c3cc(C(F)F)cs3)=O)C12 N1(C(CCCNC(C)=O)=O)CC2ON=C(CNC(=O)CC34CCCN3CCC4)C2C1 C1(C)(C(N2CC(CNC(C3(COC)COC3)=O)OCC2)=O)CCS(=O)(=O)CC1 CC1(C(=O)NC2CC2CNC(c2ccc(C3CCCCC3)cc2)=O)CCCCC1 C(c1cncc(O)c1)=CC(=O)NCCC1CCN(C(=O)CC2CCCC(=O)N2)C1 C1(NC(CCOCC)=O)CCCOC12CCN(C(=O)C=Cc1cscn1)CC2 N1(C(CC(=O)OCCC(C)C)=O)CC(F)CC1CN(C)C(C1CC1(F)F)=O CC1(C)CCN(C(=O)CCc2ccc(Cl)s2)CC1CNCC1CC2CCC1C2 Cc1c(C(=O)N(C)CC2CN(C(=O)CN3CSCC3=O)CCO2)ccn1C1CC1 C1(C(=O)NC2CN(C(CCNC(=O)OC)=O)C(C)C2)CC(C)(C)OC1(C)C C(CCCCCC1CC1)NC(c1ncn(CCNC(CC2ON=C(C)C2)=O)c1)=O O(N1CCC(CC(=O)NC2CCN(C(=O)CC3CCC(=O)C3C)CC2)CC1)CC N1(C(c2n(C)nnc2)=O)CC(O)CC1CNC(=O)CCS(C)=O C=C1CC2(C1)CC(C(N1CC(NC(C3(CC)CCCCCC3)=O)CC(O)C1)=O)C2 c1(C(=O)NC2CCCC(CNC(c3ccc(CC)s3)=O)C2)cc2c(nn1)CCC2 Cc1cc(Cl)c(C(N2CCOCC(NC(C3OCCCO3)=O)C2)=O)cc1C CN1CCN(C(N2CCC=CC2C(N2CC(OC(=N)O)C2)=O)=O)CC1 C(=O)(C(C)O)N(CCOC1(CC(=O)NC)CC1)C(C)C.C1(COC(C)=O)CC1C N1(C(C(C)(C(C)C)OC)=O)CC(CO)C2(C1)CN(C(c1cn(C)ccc1=O)=O)C2 C1(C(N2C(COC)C=CC2)=O)CC(F)CCN1C(=O)C(CO)N(C)C C1(C(=O)NC(COC)(C)C)CCC(C)(C)N(C(=O)C(C)S(C)(=O)=O)C1 N#Cc1ccc(C(=O)NC2CC2NC(=O)C2=CCCCC2)cc1C(F)(F)F c1(C(N2CCC(CN(C(COCCC=C)=O)C)C2)=O)cncc(N)c1 C1(CNC(C(C)SCCCC)=O)C(C)CCCN1C(c1ccnn1CCOC)=O C1(C(=O)NCC(CC)(C)CO)N(C(=O)CCN2CCOC2=O)CC12CCCC2 CCCCC(COC)NC(C1CCCN(C(c2nccn2C(C)C)=O)C1)=O N1(C(c2n(CCC)ncc2)=O)CCC(O)(C(C)NC(C2CCCN(C)C2)=O)CC1 C(=O)(C(C)N(C(=O)CCOC1CC1)C)N(C(C#C)C)C c1(NC(=O)NC(CCN(CC)CC)C)cc(O)ncc1Br C1(c2onc(C(C)SCC)n2)(NC)CCN(C2CC2)C1 c1(C(=O)NC2CN(C(C(CC=C)(C)C)=O)CC2O)ccnc2ccnn12 C1(NC(c2[nH]cc(CC)c2)=O)CCN(C(c2csc(C3CC3)n2)=O)CC1(C)C CC(C)C(O)C(=O)NC1(CNC(c2cc(O)cs2)=O)CC1 C(=O)(CCCCC(C)=O)N(CCC(=O)NC(CC)CO)C(C)C N1(C(COCCCC#C)=O)CCCC(NC(=O)CCc2nc(CC)no2)C(F)C1 c1(C(=O)NCC2(C)CCCN2C(=O)CC2(O)CCOC2)cccc2sncc12 CCCCCCC(=O)NC(CNC(c1nn(C)cc1C(C)=O)=O)C1CC1 C1(OC)CCCCC1C(=O)N(C1CN(C(C2CSCN2C)=O)C1)C N1(CC(C)C)CCC(C(=O)NC2CCN(C(C3(N=[N+]=[N-])CC3)=O)CC2)CC1 c1(C(=O)NC2CC(c3cn(C(CC=C)CC)nn3)C2)cc(C#N)ccc1C c1(C(=O)NCC2CCC(NC(=O)COC3CC=CC3)C2)ccc(F)c(C(F)F)c1 C1(NC(CCSCC(N)=O)=O)CC2CCC1C(NC(C1CC3(C1)CC3(F)F)=O)C2 C1(CNC(c2cnn(C)n2)=O)N(C(C2CN=C3N=CNN3C2)=O)CCCC1(C)C C1(CC(=O)NCC2CCCN2c2ccncn2)CCCOC1 c1(C(=O)NC2CN(C(CN(C)C)=O)CC2F)n[nH]c2ccc(Cl)cc12 Cc1ccc(NC(=O)CN(C)CC2CCCN2C(=O)C(O)C(C)(C)C)cc1C N(C(C(=O)NC1CC1CNC(=O)CCC1CC1(Cl)Cl)=Cc1cccs1)C(C)=O c1(COC)nc(C(N2CCC(C(F)(F)CO)C2)=O)cs1 c1(C(N(C2CCOCC2)C(C)C)=O)cnc(-c2nc(-c3ccccc3)cs2)cn1 CCCCC(C)(F)C(=O)NC1CN(C(c2ccc(OC)s2)=O)CC(C)(C)C1 N1(C(c2n(C)nc(O)c2)=O)CCN(C(=O)CC2CSCCS2)C(C(F)F)C1 c1(OC)cncc(CCC(=O)NC2CCCC2(C)CNC(=O)COCCCF)c1 c1(C(=O)NC2CC3(C(NC(C(C)n4cncn4)=O)C3)C2)cnc2nccnc2c1 c1(N2C(c3ccc(C)cc3)COCC2)cc(Br)ccc1S(=O)(=O)N1CCSCC1 Cc1nccn1C(C)CNCc1cnn(CC(F)F)c1 Cc1cncc(C(N2CC(C(O)C(=O)NC3CC3(C)C)C2)=O)c1 Cc1ccc(C(=O)NCC23CC(NC(c4cc(C(C)C)on4)=O)(C2)C3)c(Cl)c1 C(=O)(C(C)(C)CN(C(=O)Cn1ccc(C)n1)C)N(C)CC1(COC)CCC1 c1(C(N2CCC(C(C(=O)N(C3CC3)CC3CCOC3)F)C2)=O)ccoc1C1CC1 c1(C(=O)Nc2ccc(NC(c3cc[n+]([O-])cc3)=O)cn2)cc(F)c(Br)cc1Cl CC1CCCCCN1C(=O)CC(C)(C)CNC(=O)CCCCNC(N)=O c1(C(=O)NCCN(CCCCCC)C(C2CCCCC2O)=O)ccc(SC)cc1 C1C2=NOC3CN(CC23)C(=O)NC(=O)N1.C12(NC(N3CCCC3)=O)CSC(C1)C2 C(C(=O)NC1CC1NC(=O)C(CO)NC(=O)OC(C)(C)C)(C(C)C)OCC C(=O)(CCCCN(C(=O)CC1CCC(C)O1)C(C)C)N(CC(C)SC)C C(=O)(CC(O)CNC(=O)CC1CC(N(C)C)C1)NCC1(CC=C)CCCC1 CCC(CC)CC(=O)NCCCCNC(c1c(Cl)cnn1C1CCCC1)=O N#Cc1ccc(C(=O)NCCCNC(=O)CCC2CCOC2)cc1Cl Cn1ncc(C(=O)NC2CCC(F)(CNC(=O)CS(C)(=O)=O)C2)c1Br Cc1c(C(=O)NC2CS(=O)(=O)CC2NC(=O)C(Cl)=CCl)cccc1F C1(CNC(CC(CC)SC)=O)CCCN(C(=O)C(C)(C)OC(C)C)CC1 CCCCCCC(C)C(=O)N1CC(OC)CC(NC(c2cc3scnc3[nH]2)=O)C1 C1(NC(C(COC)(C)OC)=O)CC2(CCCCN2C(c2nn(C)cc2C)=O)C1 N1(C(c2ccc(CCC=C)cc2)=O)CCC(NC(=O)C(C)CCC)C12CCC2 N1(C(C(c2ccc(Cl)s2)C)=O)CCC(CNC(C2CCNC2=O)=O)C1(C)C CCC(CCC(=O)N1CCCCC1CCCNC(=O)CC1(c2ccon2)CC1)OC CC1CN2CCN1CC2C(N1CCC2(NC(=O)CO)CCCC12)=O C1(C(N(C)CC2CC(F)C2)=O)C2CCC(C2)N1C(=O)CC(=O)NC1CC1 CCCC(C)CCCC(=O)N(C)CCC1CCN(C(=O)C(C2CC2)OCC)CC1 C1(NC(c2c(C)ncn2C)=O)CCC(O)CN(C(C2CCCN(C(N)=O)C2)=O)C1 N1(C(C2CCC2CF)=O)CC2CCN(C(=O)CCCC3CCCC3)C2C1 c1(C(N(CC(CN(C(C(CC)C(=O)OC)=O)C)O)C)=O)c[nH]c2cccc(C)c12 Cc1cccc(C(=O)NC2(CNC(c3ccc(C)n3C)=O)CCC2)n1 Cc1ccc(S(N)(=O)=O)cc1C(=O)NCC(C(C)C)NC(C1CC1C)=O c1(C(=O)NCCC2CC(NC(c3c(C)cns3)=O)C2)cc2cccc(Cl)c2s1 CC1(C(=O)NC2CC(C)(NC(=O)CCC(=O)N3CCC(O)CC3)C2)CC2CC2C1 C1(C(=O)Nc2c(C(N)=O)nccn2)CC(F)CN(Cc2ccnc(Cl)c2F)C1 C1(C(N(C(C)CCNC(=O)COCC(C)(C)C)C)=O)CN(C)CCO1 c1(C(=O)NCC(CCCC)NC(C2(CC)CC2)=O)cc(F)c(OC)cc1Br c1(C(=O)NCCCN(C(C(C(C=C)C)C)=O)C)cc2ccc(F)c(F)c2o1 c1(C(=O)NC2(C(=O)OC)CCC2)cc2cccc(-c3cc(C)ccc3OC)c2s1 N1(C(c2cncc(C)n2)=O)CCCCCC(NC(=O)C(C)C(F)F)C1 C#CC1(C)CCN(C(c2cn(C)cn2)C(=O)NCc2ccccc2)CC1 C1(C(N2C(CN(C(C(C)(C)OCC)=O)C)COCC2)=O)CNc2ccnn2C1 CCCC(C(O)C(=O)N1CCCC(N(C)C)C1)NC(=O)CC(C1CC1)C1CC1 C(C(=O)N1CCC1(C)CC(=O)NC(c1cccc(C)n1)C)(C(C)C)NC(C)=O N1(C(C(CCC)N(C)C)=O)CCN(C(c2ccc(SC)cc2)=O)C(CC2CC2)C1 N1(C(C2(C)CCCCO2)=O)CC2CCCCC2(NC(c2ccc(N)cn2)=O)C1 N(C1CC(=O)c2ccccc21)C(=O)NCC1(C(=O)OC(C)(C)C)COC1 Cc1c(C(=O)NCC(C)CNC(C2CC2F)=O)cncc1F O=C(C#CC1CCCC1)NCC1CN(C(=O)Cn2cc(C3CC3)cn2)C1 c1(C(=O)NC(C(C)C)CNC(c2ccnc(Cl)c2)=O)ccc(Cl)nc1Cl N1(C(C2(C)CC=CCC2)=O)CC2CCN(C(c3cn(CC(N)=O)nn3)=O)CC2C1 c1(C(=O)NCC(c2ccc(F)cc2)(C)O)cc2cc(Br)cc(F)c2o1 CCC(CCCC(=O)OC)NC(c1cccs1)C1CCCC1 O=S(=O)(c1cccc(Cl)n1)N1CCN(Cc2cc(C(F)(F)F)cc(F)c2)C2CC12 C1(CC)CCCC(C(=O)NCC2(C(C)NC(c3ccc(O)cc3)=O)CC2)C1 C(=O)(C#CC1CCOCC1)NCC(C)(CO)NC(c1cnc(OC)s1)=O C(=O)(C(C)(C)CC(=O)OC)NC(CCC(=O)NCC1(CC)CCC(=O)N1)C CC1CN(C(=O)CCN2CCSC(C)(C)C2)CC(C)C1NC(=O)C=CC(C)(C)C c12cc(ccn1)NC2=O.C1(C(=O)NC2(C)CC(C(=O)OC)C2)C2CCC(=O)C12 c1(C(=O)OCC)cc([N+](=O)[O-])c2c[nH]nc2c1.c12nnnn1CCS2 N1(C(C(CC2CCC2)OC)=O)CCC2CC2(C(=O)NCC2CC3CC3C2)CC1 N1(C(CC2N(C)CCC2)=O)CCc2cc(CNN3CCOCC3=O)ccc2C1 C1(CC=C)(NC(=O)CC(C)C)CCN(C(=O)Cc2ccc(-c3nc[nH]n3)cc2)C1 N1(C(C2(C=C)CCOCC2)=O)CCCC(C2CCN(C(C3(C)CC3C)=O)CC2)C1 N1(C(=O)NC)CCC(C(N2CCC(CF)(NC(c3cc(C)sn3)=O)C2)=O)CC1 CC1(C(=O)Nc2ccc(OC(F)(F)F)cc2Br)CCN(S(C)(=O)=O)CC1O C1(O)(CNC(C2C(CNC(CCN(C)C3CC3)=O)C2)=O)CCSCC1 CC(C(=O)NC1CC1)=C1CN(C(=O)C(=O)NC2(CO)CCC2)C1 c1(C(N2CC(OC)C(NC(=O)CC3CC3(Cl)Cl)C2)=O)csc2ncnc(O)c12 N1(C(=O)Nc2c(OCC)nn(C)c2)CC(C)(CSC)CC1(C)C c1(N2CC(CN(C(=O)CSC(F)(F)F)C)OCC2)ccc([N+](=O)[O-])c(C#N)c1 N1(CCNC(c2c(OC)c[nH]n2)=O)CCN(C(c2scc(C)c2Cl)=O)CC1 N1(C(CNC(CCC)=O)=O)CC=CC(NC(C2(O)CCSCC2)=O)C1 C(C(C)(C)C(C)(C)C)NC(C1(COC)C=CCN1C(c1ccnc(OC)n1)=O)=O n1(CC(=O)NCC2CC(C)N(C(c3ccc(O)c(N)n3)=O)C2)cc([N+](=O)[O-])cn1 N1(C(c2nc(CC)oc2)=O)CCCN(C(=O)CC2(C#N)CCC2)CC1C C1(C)(CCCC)NC(=O)N(NC(=O)c2sc3c(c2Br)CN(C(C)COC)C3)C1=O S(=O)(=O)(c1cccc(N2CCCC3(CCCC3)C2)n1)N1CC(C)C(C)C1 CN1CCC2CCN(C(c3cccc(OCc4ccccn4)c3)=O)CC2C1=O S(=O)(=O)(c1cnn2ccc(=NC(C)C3CCOC3)[nH]c12)NCCSCCOC Cc1nn(CCO)c(C)c1C(=O)N(C)CCN(C)C(C1CN(C(N)=O)C1)=O C(=O)(CCC(C)(C)[N+](=O)[O-])NC1C2CC(C(N3C(C)(C(=O)NC)CC3)=O)C(C2)C1 c1(C(=O)NC2CCOC(c3cccnc3)C2)c[nH]c2ncc(Cl)cc12 N1(C(COCc2n(C)ncc2)=O)CCC(C2(NC(=O)C3=COCCC3)CC2)C1 N1(C(C23CC(OC)C2C3)=O)CCC(CNC(=O)C=CC(=O)N(C)C)(OC)CC1 CCC(C)(O)C(=O)N1CCC(N(C(=O)CN(C2CC2)CC)CC2CC2)C1 c1(C(N2CC(C)(NC(=O)C3=CCS(=O)(=O)C3)C2)=O)ccc(O)c([N+](=O)[O-])c1 CC#CC1CCN(C(C23C(NC(=O)C(F)C4CCCC4)C4CC2C3C4)=O)C1 C(=O)(C(C(C)C)NC(c1n[nH]c(=N)[nH]1)=O)N(CCCC(=O)NC)C Cc1cc(NC(=O)CN(C(=O)C(C2CCC(=O)N2)C)C)cc(O)c1 Cc1cc(C(=O)N(CCNC(C2CC3CC3C2)=O)C(C)C)c(F)c(Br)c1 C1(C(=O)NC2(CC=C)CCN(C(c3cccnn3)=O)C2)CCc2nccn2C1 c1(C2(CNC(c3c(C(=O)OC)nccn3)=O)CC2)ccc2c(c1)OCO2 N1(C(C2(NC(=O)CCC=C(C)C)CC(=C)C2)=O)CCCN(C2CC2)CC1 C(=O)(C1=CC2CCCC12)NC1(C)CCN(C(CCC=C(C)C)=O)CC1 C(=O)(C1=CCC(C)CC1)NCCC1(O)CCCN(C(c2cc(OC)nn2C)=O)C1 c1(C(=O)NC(C(=O)NCC(CC2CC2)CO)C2(C)CC2)cccnc1O C(CN=C(NCC(c1ccncc1)C)NCC(C)C)OCC Cc1ccc2c(c1)C(C(=O)NC(CNC(c1cc(C)c(F)cn1)=O)CC(C)C)C2 C(=O)(CCCCCCN=[N+]=[N-])NCC(CC)NC(c1cnn(CC)c1C1CC1)=O C#CCCC(O)C(=O)NCC1CC(CNC(C2(CC#C)CCCC2)=O)C1 N#Cc1ccc(C(N2C(C(=O)NC3C4COCC34)CCC2C2CC2)=O)o1 O(NC(=O)C(F)C(C)C)C(CC(C)C)C(=O)N1CCN(C(C)C)CC1 C12C=CCC(C1)C(=O)Nc1cn2nn1.C(CCC(=O)NC(C)C(=O)OC)N(C)CC C(C(=O)NOCC(F)F)(C1CN(C(c2ccc(C)o2)=O)C1)OC c1(C(=O)NC2C(NC(c3c(C)nc(C)[nH]3)=O)COCC2)cnn2c1CC(F)(F)C2 Cc1cc(C(=O)NC2CN(Cc3ncccc3Cl)CC2C#N)c2cc[nH]c2c1 c1(C(=O)NC(C(C)NC(C2C(C)C2C)=O)CO)c(F)cc(C#N)cc1F C1(NC(CCc2ccc(SC)cc2)=O)CCN(C(c2ccccc2Cl)=O)C12CC2 C12CN(CC13CCC3)C2=O.C1(C(N2CCCC(C(=O)O)C2)=O)CC2CCCC2C1 N1(C(CCNC(COC)=O)=O)CC(CC(=O)NCc2cn[nH]c2)C2(CC2)C1 c1(NCc2c(C)cc(N)cc2)[nH]c(=NC2CC3CC3C2)nc2sccc12 CC(CN(C(=O)CC1CCCOC1)C)C(=O)NC(c1ccnn1C)(C)C N1(C2CCN(C(C(C)OCC=C)=O)C2)CCN(C(c2nc(CC)sc2N)=O)CC1 c1(C(N2CCC(CC=C)(NC(c3nccn3C)=O)C2)=O)cnc2cccnc2c1 N1(C(C2C(C)(C)CC2)=O)CC2CC2(CNC(=O)C(c2ccc(F)cn2)(F)F)C1 c1(NC(CN2CCC(C)C2)=O)cccc(CNC(=O)CCc2nc[nH]n2)c1 c1(C(C(=O)OC)NC(=O)NCc2cc(C(C)C)on2)cccc(C(F)(F)F)c1 C(C#Cc1ccccc1Cl)NC1CCN(C(C2CC2c2cccc(Cl)c2)=O)C1 C1(C(=O)NCC2(F)CCCN(C(CSCC)=O)C2)CCC(F)(F)CC1(C)C c1(C(N2CCN(C(C(C(C)C)OC)=O)CC2)=O)ccc2ccc(C)cc2n1 c1(C(=O)NC(CCNC(Cc2c(F)ccc(C)c2)=O)(C)C)n[nH]c2c1CSCC2 N1(C(CC(CNC(C(C)OCOC)=O)C2CCC2)=O)C2CCCC1CC2 c1(C(=O)NC2C3CN(C(C(F)=CCC)=O)C2C3)c(O)cc(=O)n2c1COCC2 c1(CCC(=O)NC(CNC(C(COCC)C)=O)CO)ccc2nc(O)[nH]c2c1 c1(C(=O)NCCCOC2CCN(C(C3CCCO3)=O)CC2)cc(F)cc(Cl)c1N C1(NC(COCCCC(C)C)=O)CN(C(C2(c3cc[nH]n3)CC2)=O)CCC1CO N(C)(C1CCc2ccc(OC)cc21)C(N1C(c2onc(CC)n2)CCCC1)=O c1(C(=O)NCCC(=O)NCC(CO)NC(=O)Cc2ccco2)cc(Cl)ccc1Cl C1(CNC(C2C(C)C2C)=O)CCN(C(c2cc3ccncc3s2)=O)CC1(F)F C1(CNC(c2c(C)ocn2)=O)CC2(CC2)CN1C(c1cncc(F)c1C)=O C1(C(=O)NC2CCC(N(C(=O)CCN(S(C)(=O)=O)C)C)C2)OC(C)(C)OC1(C)C C1(C(=O)NCC2(SC)CC2)CCC(C2CC2)N1C(=O)CCC1(C)CC1 c1(C(=O)NC2C3CN(C(CCOCC)=O)C2C3)oc2c(Br)cccc2c1C CCC(C(C)CN(C)C)NC(=O)CC1CCCN(C(=O)C(COC)N(C)C)C1 C12(NC(C3CCC(OC)C3)=O)CC(C(F)(F)F)C1CN(C(=O)C(F)=CCCF)C2 NC1CC2(C1)C(C(N1CCC(CCN3CCCCC3)CC1)=O)C2(F)F c1(C(N2CC(=O)OCC2)=O)cc(F)cc(Br)c1F.c12csc(n1)NC(=O)C2 C12(C(N(C(C)C(N)=O)C)=O)CC(NC(=O)CC3OCCCO3)(C1)C2 c1(CCC(=O)N(CC(C)NC(C2CC2(C)C)=O)CC)ccccc1 c1(OC)cc(C(N2CCC2C(=O)N(C(CO)CO)C(C)C)=O)ccc1OC(C)=O N1(C(C(=O)NCC2CCCCC2(F)F)=O)CC2CC(c3cc[nH]n3)C2C1 Cc1cc(=O)n(C)nc1C(=O)NC(C)CN(C)C(c1c(C)nn(C)c1Cl)=O Cc1cc(C(=O)NC(C)CCNC(=O)CCNC(c2cccs2)=O)ncn1 c1(C(C)C)ccc(CC(=O)NCCC(O)CNC(=O)C=C2CCOCC2)cc1 c1(CC)noc(C)c1C(N1CC(CNC(C2CC(N=[N+]=[N-])C2)=O)C(C)C1)=O C(=O)(CCC(=O)N1CCC(c2ccccc2)=N1)N(CC(COC)O)C c1(-n2ncc(C(N(CC(C)N(C(CC=C(C)C)=O)C)C)=O)c2)ccccc1C C1(C(=O)NCC(C)(C)Cn2cc(C3CC=CCC3)nn2)(OC)CC(C)(C)C1 C1(COC)CN(C(=O)C=CC(=O)N(C)C)CCN1C(C1CCC(F)CC1)=O C1(COC)CN(C(C2CC2C(F)(F)F)=O)CCN1C(=O)Cc1nc(C)no1 c1(COCC(=O)OC)ccc(C(=O)NCC2CCCC2)nc1.C1(=O)CSCCN1 n1(CC(=O)NC2(c3ccc(=N)[nH]c3)CC2)ncc2cccnc12 C(C(O)CCNC(=O)CCCOCC)NC(COCC)=O C1(C(=O)NC(C2CCN(C(=O)CSC(C)(C)C)C2)C)COCCOC1 n1(CC(=O)NCC(C)(CO)NC(C2CN(CC)C(=O)C2)=O)cc(Cl)c(O)nc1=O Cc1noc(C)c1S(=O)(=O)NCC(=O)N(C1CN(C(C2CCCS2)=O)CC1O)C c1(OCC(=O)N(CCNC(C2CC23CC(O)C3)=O)C2CC2)c(Cl)cccc1Cl Cc1ccn2ncc(C(N3CCC(CNC(c4ccsn4)=O)CC3C)=O)c2n1 C1(NC(C2(CC=C)CCCN2C(=O)C(O)C2CC2)=O)C(O)C2CCOC12 Cc1cc(C)c(C(=O)NC2CCN(Cc3ncccc3Br)CC2F)c(Cl)n1 C(c1ccc(F)c(Cl)c1)=CC(N1CCN(C(C2C(C=C)CC2)=O)C(CCO)C1)=O N1(c2cc(NC(C)CCN3CCCC3)ncn2)CCC(O)C(F)(F)C1 c1(NC(CN(CCC(=O)N(C(CC(CC)C)C)C)C)=O)ccc(Cl)cc1F N1(C(NNC(c2cccc(C(=O)OC)n2)=O)=O)CCCC(C)(C#N)C1 Cc1oncc1C(=O)NCC1(O)CC(CNC(=O)CCCn2ccnc2C)C1 c1(C(=O)NC2(CNC(c3c(C)nc(O)s3)=O)CC2)ccc([N+](=O)[O-])s1 C1(C(N(C2CN(C(c3c(Br)cc(C)c(F)c3)=O)C2)C)=O)CCc2ccccc2C1 C(C)(C)(CCCC(=O)NCc1ccc(C#N)cn1)NC(CC(CN(C)C)O)=O C1(NC(Cn2c(C)nc(C)n2)=O)CC(C)CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)C1 C1(CNC(=O)CN2CSCCSC2)CC2(C1)CN(C(c1ccncc1)=O)C2 Cn1cc(C(F)=CC(=O)NCC2CN(C(C3(Cl)CC3)=O)CC2(C)C)cn1 Cc1ccc2occ(C(=O)NC3CC(NC(=O)C(F)=C4CCCC4)C3)c2c1 C(=O)(C(O)C(F)(F)F)N1C(CNC(C2CN(C)CCN2C)=O)CC(COC)C1 N1(C(c2cccc(C#N)c2)=O)CC2CN(C(c3cc(O)no3)=O)CC2C1 C1(C(N2CCN(C)CC2CO)=O)COC2(C1)CN(C(=O)C#CC1CCC1)C2 c1(CC(N2CCC(F)(CNC(CCCOCCC)=O)C2)=O)cc(OC)cc(Cl)c1 N1(C(C)C)CCn2nnnc2C1.c1(OC)cccc2c1NC(=O)NCC2 C1(NC(C2CN(C3CCOC3)C2)=O)CN(C(C2C(Cl)(Cl)C23CC3)=O)CCC1O Cc1cccc(C(N2CC3CC(NC(=O)COCc4nccn4C)C2C3)=O)c1N c1(C(=O)NC2(C)C(C)(C)CCCC2)ccccc1S(=O)(=O)NC(C)(C)C C1(NC(c2ccc(C(C)C)o2)=O)CCCC(N(C(=O)Cc2cn(C)nn2)C)C1 c1(C(N2C(CNC(=O)CCn3cncn3)CC(OC)C2)=O)ccc(C)nc1O N1(C(C)=O)CCC(C(=O)NC(C)(C)CNC(c2coc(O)n2)=O)CC1 C(=O)(C1COc2ccccc21)N(CCC(C)(C)NC(C1CCC2CC2CC1)=O)C Cc1cc(NC(N2CCCCC2)=O)ccc1OC(F)F.C1C(=O)N1 S(=O)(=O)(c1cccc(C(N2CC(C)(C)C2C(=O)O)=O)c1)NC(CC)C Cc1ccc(SCC(C)NC(C2CC(CC(C)(C)C)C2)=O)cc1 S(=O)(=O)(C1Cc2ccccc2C1)N(C1C(C)CCNCC1)C1CCCCC1O O=C1CCC(C(N2CC(c3ccccc3)(NC(c3ccccc3)=O)C2)=O)CCO1 c1(C(N2CCC(C)(CN(C)C)C2)=O)c(Cl)cccc1I c1(C(N2CCC(N(C(CC(C)c3ccco3)=O)C)C2)=O)cc2cccn2c(O)n1 C#CCC(CO)NC(=O)C=CCN(C)C(C1(N(C)C)CCC1)=O CS(=O)(=O)c1nccc(N2CCC3CN(Cc4ccc[nH]4)CC23)n1 C1(NC(=O)Cc2ccno2)(CNC(c2n[nH]c(C3CC3)n2)=O)CCOCC1 c1(-n2c(COC)ncn2)ccc(C)c(Br)c1.CC CC1Cc2ccccc2N2C(=O)N(C3CCC(c4ccc(Cl)cc4)C3)C(=O)C12 C1(C)(CC)C=C(C(=O)N2CCN(C(C3COC4(CCC4)C3)=O)CC2)C1 C1(C)(N)CN2CCC1CC2.C(CCC(C(=O)OCC=C)NC(=O)OC(C)(C)C)=C(C)C C1(C(N(C(C)C)CCNC(=O)C(C)Cc2ccncc2)=O)COC2(CCC2)CO1 C1(F)(C(N(CCCOCCNC(C(C)OCCC(C)C)=O)C)=O)CCCC1 n1(CC=C)c(N(CCC)CC)nnc1CCc1ccccc1 n1(CCCNC(=O)NC2CC3COCC3C2)cc(Br)ccc1=O N1(C(c2cncc(C)n2)=O)CCN(C(=O)C(C2CC2)C2CC2)CC12CCC2 c1(OC)cnc(F)cc1C(N1CC(NC(C2COC2)=O)C(c2ccccc2)C1)=O c1(C(=O)NCC2CN(C(CCSCC)=O)C(C)CC2)ccc2c[nH]nc2c1 c1(C(=O)NC2CCN(C(C(COCC)C)=O)C2)c(C(F)(F)F)noc1C CC1(CNC(=O)CO)CCC(NC(c2occc2-c2ccccc2)=O)CC1 CC1CC(CNC(=O)Cc2cnc[nH]2)CN1C(=O)Cc1ccsn1 c1(C(=O)NC2CN(C(c3[nH]cc(C)c3)=O)CC2C)cc(O)c2c(C)nn(C)c2n1 N1(C(C(F)=C(C)C)=O)CC(O)CCC1C(=O)NCC(C)(C)C(C)(F)F c1(OC)ccncc1NC(C1(C2CCCN2C(c2cc(C)oc2C)=O)CC1)=O c1(CNC(c2ccc(NCC3CC3)cc2)=O)c(F)cc(Cl)cc1F C12(C(=O)NCc3ncc[nH]3)CCN(C(c3ccc(F)cc3F)=O)CC1C2 CC1CCCC=C1C(=O)N1CCCC(NC(=O)Cn2cnc(Br)n2)CC1 N1(C(Cc2c(SC)cccc2)=O)C2CCC1CN(C(=O)COc1cc(C)on1)C2 N1(C(CCC=CCC=C)=O)CCC2(CC1)CC(NC(=O)C(C1CCCCC1)C)C2 Cc1ccc(C(=O)NCC(O)CC(=O)NC(C)CC2CCCCC2)c(C)c1 CC(CCS(C)(=O)=O)Sc1ccc(NC(=O)C(N2CCC(N)CC2)=O)cc1 CC(CC(C)NC(=O)C(c1ccc(N(C)C)cc1)C)N=c1nc[nH]s1 O=C1CCn2nc(N3CCC(NC(=O)NCCc4ccnc(Cl)c4)C3)cc21 C1(C(=O)NC2(CC(=O)NC(C(C)C)(C)CO)CCC2)CCCCCN1C C1(CC#C)(C(=O)N(CC(CO)(CO)NC(C2CCCCC2O)=O)C)CCCOC1 c1(C(=O)OC)cc(=NC(=O)C(=O)NCCc2ccsc2)[nH]n1C C1(CNC(c2n(C(C)C)ccn2)=O)C(C2CC2)CCN1C(c1cnc[nH]1)=O c1(C(=O)NCC(C2N(C(c3c(C)cnn3C)=O)CCC2)(C)C)cc(O)nc(O)n1 N1(C(C(C(C)C)CNC(c2cccs2)=O)=O)CCC2(C=CCO2)CC1 c1(C(=O)NCC23CC(NC(c4c(C)nc(C)o4)=O)(C2)C3)ncnc2ccsc12 C1(CNC(C2CN(C(N)=O)C2)=O)CC2(C1)CN(C(C1CCC=CCCC1)=O)C2 C1(C(N2C(C)C(NC(c3cn(C4CC4)nn3)=O)CC2)=O)CC2(CCC2O)C1 O=NN1CCCC1C(=O)NCC(F)CNC(=O)Cc1csc(-c2ccccn2)n1 N1(C(C(C)OCCOC)=O)CCC(C(C)CNC(c2ncn(C)c2C)=O)CC1 c1(C(=O)NCC2(F)CN(C(c3cnc(CC(C)C)[nH]3)=O)C2)cccc(Cl)c1F C1(NC(c2cnns2)=O)C(CNC(C2CC(Cl)(Cl)C2)=O)CCC12CCC2 N1(CC=C)CCN(C(=O)NCc2cc3cscc3s2)CC1=O c1(NC(c2c(C)nccc2)=O)ncccc1[N+](=O)[O-] C(C)(C)(C(=O)N(C1CC(NC(=O)CN2CC3CC3C2)C1)C)OC(C)C N1(C(c2c(CCC)[nH]cc2)=O)CCn2ncc(S(C)(=N)=O)c2C1 C1(C(=O)NC2CC(CNC(C3CCC3)=O)C2)CCCN1C1CC1 c1(C(=O)NC2C(CNC(c3cc(C)n(C)c3C)=O)C2)cccc2c1CC(C)(C)C2 N1(C(C(CSC)C)=O)CCCC(CCNC(c2cccc(-c3nnco3)c2)=O)C1 N1(C(=O)Cc2csc(NC)n2)CC2CCN(C(=O)C3=NOCC3)C(C2)C1.NC=O c1(CN2CCC(C(=O)NCCC)C2)ccc(CCC)c(Cl)c1 c1(CC(=O)NC2CCCN(C(C3(F)C(C)C3)=O)C2)ccc2nc(O)[nH]c2c1 C1(OC)CN(C(c2ccn(C)n2)=O)CC1NC(=O)Cc1cc(C)[nH]n1 c1(CC(=O)NCC(=C2CN(C(CCN(CC)CC)=O)C2)F)cccc(C)c1Cl N1(C(c2c(CC)con2)=O)CC2CCC1CC2NC(c1c[nH]c2nccc-2c1)=O C(=O)(CCCN(C)N=O)NC1(COC)CC1.C1(=O)CC(C)N1.C1(C=O)CCCCC1 Cc1n[nH]c(C)c1-c1ccc(C(=O)NCC2CC(NC(=O)CN(C)C)C2)cc1 c1(NC(C)=O)ccc(C(=O)NCC(O)CN(C(=O)C=C(C)C(C)C)C)c(F)c1 C(C(=O)NC(C1CN(C(=O)Cc2cc(C3CC3)on2)C1)C)(C(C)(C)C)SC c1(C(=O)NC2(C)CCC(NC(CC(C)OC)=O)CC2)cccc2c1OC(C)(C)C2 S(=O)(=O)(C(F)(F)F)ONC(c1nc(C(F)(F)F)cs1)=O.S(C)(=O)(=O)N CCCCCC(C)CC(=O)NCC(C)CN(C)C(c1ccncc1)=O Cc1ccc(C2(F)CN(C(C3C(C)C3C)=O)C2)cc1 CC1=C(C(=O)NC(C2CCOC2)CNC(c2cnc(O)n2C)=O)COCC1 Cc1nnc2n1CCC(C(=O)NCC1(CNC(=O)CCCCCC(C)O)CC1)C2 N1(C(Cc2cc(C)nn2C)=O)CC2(C)CC1(C(N1CCC(F)(C#N)C1)=O)C2 Cc1cc(C(N2CCCC(N(C(=O)CC(C)O)C)C2)=O)cnc1C(F)(F)F c1(CC)onc(C)c1C(N1CC2(NC(C3CC3(F)F)=O)CC1C2)=O c1(C(=O)NCC)ccc(S(=O)(=O)NCc2ccc(OC)c(Br)n2)cc1 C1(C(C)(C)O)CCN(C(C2(CNC(=O)C(O)C3CC3)CC23CCC3)=O)CC1 N(C1c2ccccc2OCC1O)C(=O)NCc1csnn1 C(=O)(CCCCN1C(=O)CCC1=O)NC(CCN(C(C(C=CC)O)=O)C)C C(=O)(CCC(F)(F)C(F)(F)F)NCC(C(C)C)NC(c1scc(OC)c1)=O c1(C(=O)NCC(C)N(C(=O)Cc2ccsn2)C)cc(N)ccc1Br C1(NC(Cc2nc(C)c(C)s2)=O)CCCN(C(c2c(C(C)C)cnn2C)=O)CC1 c1(N2CCC(NC(=O)CCc3nc[nH]n3)C(F)C2)nc2c(cc1Cl)C(=O)OC2 c1(-c2cn(C3CN(C(C(c4cccnc4)OCC)=O)C3)nn2)cc(C#N)ccn1 C1(C(=O)NC2(C(=O)N(C3CCCC3(C)O)C3CC3)C(C)C2)CC(C)(C)CCO1 C(C1(F)COc2ccccc21)Nc1c(OC(=O)OC(C)(C)C)cc(Cl)c(Br)c1 C(C)(C(=O)NC(C1CN(C(=O)CN(C)C2CC2)C1)C)OCC=C CC(C)(C)CC(F)C(=O)N1CCCCC1CNC(=O)CCNC(=O)CC(C)(C)F Cc1cccnc1C(N1CC(CNC(c2cnncc2C(F)(F)F)=O)C2CC12)=O N1(C(C(C)SC)=O)CC(NC(=O)CCCc2ccc(F)cc2)CC2(CCC2)C1 Cc1ncnc(C)c1C(=O)NCC12CC(CO1)N(C(c1ccnc(CO)n1)=O)C2 N1(C(C2C(=C)C2)=O)CCN(C(=O)C(=O)N(CCOCCO)CC)CC1 C=CCC(CC)C(=O)N1CCCC1CCC(=O)NC(c1nc(C)no1)C C1(CCC)CCCN(C(C2CC=CCC2CN)=O)CC1 c12ccc(cc1)COCCN2CC.c1(C(=O)OC)nc(Cl)sc1Br C1(C(=O)NC(C)C(C)(C)NC(c2ccc(CF)cc2)=O)CCCC2(CC2)C1 c1(C(=O)OC)ccnc(NCC2CN(C(c3coc(C)n3)=O)CC2C(F)(F)F)n1 C1(CNC(C(C(C)C)OC)=O)CN(C(c2cc(C(F)F)nn2C)=O)C2(CCC2)C1 CC(CN=c1[nH]c2c(c(=NCc3cn(C)cn3)[nH]1)SCC2)C1CCC1 O=C1CC(=O)NC(C(=O)NCc2nocc2C(N2CCCCC2CF)=O)C1 CC(CF)CC(=O)NC1CCCC(NC(=O)CN2CCC(O)CC2)C1 CCC(C)C(C(=O)NCC(C1CCC1)OC)N(C(=O)CCc1csnn1)C N1(C(C(C(=O)OCC)F)=O)C2CCC1CN(C(=O)CCC=Cc1ccccc1)C2 C=CCCCCC(=O)NC(CCCC)C(=O)NCC1(C)C=CCCC1 C1(CC(=O)NCC(C(C)O)C)(CC(=O)O)CS(=O)(=O)C1 c1(C(=O)NC(C(CO)NC(COCC=C)=O)C)cccc2c1CCOC2 c1(C(N(CCCNC(c2cc(C)on2)=O)CC)=O)cnc2c(c1)CCC(=O)N2 C1(CC)C(NC(C2(n3nccn3)CC2)=O)CCN1C(c1ccc(C2CC2)s1)=O c1(CC(C(C)C)NC(C2(S(C)(=O)=O)CC2)=O)ccccc1F c1(SCC(=O)N(CC)CC2N(C(C(C)n3cccc3)=O)CCC2)cccc[n+]1[O-] CS(C)(=O)=NCC(=O)N1CCC(CNC(=O)C(C2CC2)NC(=O)OC(C)(C)C)C1 N1(C(C(C)OC2CCCC2)=O)CCCC2C1CCN2C(c1ccnnc1)=O C(CC(O)CNC(c1nncs1)=O)NC(=O)CCc1ccc[nH]1 N1(C(CCCC=C)=O)CC2(CC(CNC(C3CCC(C)O3)=O)C2)C1 N1(C(C(=O)C2CCCC2)=O)CC2(CNC(=O)CSCc3cccnc3)CCC1C2 N1(C(C)=O)CCC(F)(CNC(=O)CN2CCN(C)CC2)CC1 CCCCCC(O)CC(=O)N1C(C(N2CCC(C)(C#N)C2)=O)CCC1C1CC1 N1(C(C23CC(OC)C2C3)=O)CCC(NC(c2coc(C#N)c2)=O)CC1 C(CN=c1nc(N2CC3CC2CC3O)cc[nH]1)c1c(C)n[nH]c1C C1(CN(C(=O)CCCC2CC2)C)CCCN1C(=O)C(C)(C)n1cncn1 c1(N(C(C2C(CNC(CCCN(C(C)=O)C)=O)CCC2)=O)C)ccc(C)c(C)c1 c1(C(N2CCCC(NC(C3C(C=C)C3)=O)C2)=O)cc2n(n1)CCCN2 CCC(CO)CCNC(C1CC(NC(C2CS(=O)C2)=O)C1(C)C)=O C(=O)(CCCCCCNC(C1CCSCC1)=O)NCCC(C(C)C)C CC(C)CCC(=O)NCc1ccoc1C(=O)NC1C(O)CC1O C1(C(=O)NC2(CO)CC(OC)C2)C=CCN(C(=O)CC2(N(C)C)CCCC2)C1 c1(C(=O)NC2CCN(C(C(c3ncccn3)C)=O)CC2F)cc(Br)cc(F)c1F C1(C(N2CCC(N(CCC)C(C3CCCO3)=O)C2)=O)CCC(OC)CC1 C1(CC(=O)NCCOC(C)(C)CNC(C2C3CC4C(C3)C24)=O)OCCCC1(C)C CCCCCC(F)C(=O)N1CCCC1C1CCN(C(c2ccn(C)c2)=O)C1 C1(CNC(C2CCC(=O)NC2)=O)CC2(CC2)CN1C(=O)C(O)C1CCC1 CCCC(CNC(=O)CC=CC(C)(C)C)NC(c1cnn(CC)c1)=O C(=O)(C(C)CC(C)(C)C)N1CCC(O)(CCNC(c2c(C)c(N)ccc2)=O)CC1 C1(NC(C2C(S(C)(=O)=O)CCC2)=O)CCN(C(=O)C#CC2CC2)CC12CCC2 C1(=CC(=O)NC2C(NC(c3c(C)cc(CO)o3)=O)CC2)CCCCC1(C)C N1(C(CC2(C=C)CC2)=O)CCC(CC(C)NC(=O)Cn2cnccc2=O)CC1 C1(NC(CC2C(C)(C)C2(C)C)=O)CC2CC1CN(C(=O)C(O)C1CCC1)C2 c1(C(N2C(C)CC(CCNC(C3CCCCC3)=O)CC2)=O)ccn2nccc2c1 c1(CC(N2CCCC(NC(=O)Cc3ccc(Cl)cc3)C2)=O)cccc(Br)c1F c1(CC)nc(CCNC(=O)C(c2cccnc2)NC(=O)CC2CNC(=O)O2)n[nH]1 c1(N(C(CCNC(C(CC)(C)OC)=O)C)C)cc(S(C)(=O)=O)nc(C)n1 c12ccc(cc1)C(=O)OC2.C(C1CCCCC1)=CC(=O)NC(CC)CO c1(CNC(CNC2(C(=O)OC(C)(C)C)CCOC2)=O)cccc(F)c1 CC1(C)CCC12CN(C(C1CSCN1C(c1nnc(O)nc1O)=O)=O)C2 C1(C2CCC(=O)NC2)(C(=O)NC(CC(C)NC(c2c(C)ncn2O)=O)C)CCC1 c1(C(N2CCC(N(C(c3ncsc3C)=O)CC)C2)=O)noc2c1CC(F)(F)CC2 CN1N=C(C(=O)NCC2(F)CCCN(C(c3cc(Br)c[nH]3)=O)C2)CCC1=O c12cc(on1)NC(=O)C(C)(C)OC2.C(CO)(C(=O)N(C)C)NC(C)=O N1(C(CC2(OC)CCC2)=O)CCC(O)C(NC(=O)C(N2CCCC2)C2CC2)C1 c1(C(=O)NC2CN(C(CC(N3CCC(C)CC3)=O)=O)C2)cc2c([nH]1)CCC(C)C2 C(CS(=O)(=O)CC(=O)NCCCNC(=O)CN1CC(F)(F)C1)OC C(=O)(CC(=O)OC(C)(C)C)NC(C)CCNC(c1ccns1)=O Cn1cc(C(=O)NCCC2CC(NC(=O)Cc3ncc(Cl)s3)C2)n(C)c1=O N1(CC(=O)NC2C(NC(Cc3n(C)nnc3)=O)CCOC2)Cc2ccccc2C1 N1(C(C(CCCC)C)=O)CCC(C2CN(C(=O)CC3CCCCCO3)C2)CC1 c1(CC)cnc(C(=O)NCC2COCCN2C(=O)CCNc2ccccc2)cn1 C1(CNC(C2C(OCC)C2)=O)CC(F)(F)CN1C(C1CCCCC1(C)C)=O C1(C(=O)NC(CNC(c2c(COC)ccs2)=O)(C)C(C)C)Cc2nnc(C)n2C1 C=C(C)C1OCCC1C(=O)NC1CC1NC(=O)C=C=C(C)C CCCC(CC)C(=O)N1CCCC(NC(=O)CCn2cc(C)cn2)CC1 N1(C(C(CSC)C)=O)CC2CCN(C(=O)CC3(C#N)CCOCC3)C2C1 CC1OC2CCC1(NC(C1(CO)CCCN(C(=O)C=Cc3ccsc3)C1)=O)C2 C1(C(N2CC3CC3(CNC(c3cnc(C(C)=O)s3)=O)C2)=O)(COC)CCOCC1 C1(C)(CNC(C2C(=C)CC2)=O)CCN(C(C2CCCN2CCC)=O)CC1 C(CC(C)C)(C(=O)NCC1CC2CC2C1)N(C)Cc1c(SC)cccc1 C1(NC(c2cc(C3CC3)ccc2F)=O)CCCN(C(C2(F)CCC2)=O)CC1 N1(C(C(C)(C)O)=O)CCC2(C1)CN(C(=O)CC(O)Sc1ccccc1)CCO2 N1(C(COC2(C)CCCC2)=O)CCC2(CC1)CC2CNC(C1CCCC1(C)C)=O N1(C(C(C(C)C)C(C)=O)=O)CC=C(CCN(C(C2(NC(C)=O)CS(=O)(=O)C2)=O)C)CC1 Cc1cc(C(=O)NCCC2CCCCN2C(=O)C(C)Cn2ccnc2)ncn1 Cc1nccn1CCNC(=O)C(C)(C1CC1)N(C)C(C1CCC(=O)C1)=O N1(C(C(=O)NC(c2ccccc2)C)c2cscn2)CCNCC1 C1(CNC(=O)COCC(F)F)CC2CCCC2N1C(=O)CCN1CCCCCC1 CCC(C)(CNC(c1ccc(CNC(c2cc(C(F)F)[nH]n2)=O)o1)=O)C(C)O Cc1c(C(=O)O)sc2ncnc(N3CCCC(CF)C3)c12 N1(C(c2c(CC)nc[nH]2)=O)CCC2CCC(C1)N2C(c1cc2cnccc2o1)=O N1(C(C2CC(OC)C2)=O)CCC2CC1CN2C(C1CCC2CC1C2(C)C)=O C1(C(C)NC(C2CN(S(C)(=O)=O)C2)=O)CCCCN1C(c1cccc(=O)o1)=O c1(C(=O)NCC2CCN(C(c3n(C)ccn3)=O)C2)cc2c([nH]1)CCC2 c1(C(N2C(CCN(C(COC)=O)C)CCCC2)=O)ccc2c(c1)N(C)CC2 c1(CC(=O)N(C2CCN(C(C3CCCCC3F)=O)C2)CC#C)ccccc1OC C(=O)(C(CC(C)(C)C)NC(C1COCCO1)=O)N(CC(C)N(C(C)=O)C)C Cc1csc2c(N3CC4CCN(Cc5c(Cl)ccc(Br)c5F)CC4C3)ncnc12 CC(C)CCCC(=O)NCC1(NC(C2C(C)C2C)=O)CCC1 C(=O)(C(F)C(C)CNC(=O)C(C)N1CCCC1)NCc1cc(C)ns1 c1(OCC)cc(C(N2CCC(N(C(=O)CN3CCOC3=O)CCO)C2)=O)[nH]n1 c1(OCC(N2CC=CC(NC(=O)CSC3CC3)C2)=O)ccc(C(F)(F)F)cc1Cl C1(OC)CN(C(C2CCC(CNC(c3cnc(=N)[nH]c3)=O)CC2)=O)CC12CC2 c1(N)cn(C)ccc1=O.N(C=CC(=O)C(F)(F)F)Cc1n(C)cc(NC(=O)C2CC2)c1 C(=O)(CCCS(N)(=O)=O)N1CCC(CC=C)(NC(=O)C(C(C)(C)C)OC)C1 C1(C(=O)NC(CC)C(C)O)CCC(CNC(c2ccc(OC)nn2)=O)CC1 c1(C(=O)NCC(C2CC2)NC(C#CC(OCC)OCC)=O)cnc(C)nc1CC c1(CNC(C2C(C(C)C)C2)=O)ncoc1C1CN(C(=O)CNc2ccccn2)C1 c1(CNC2C=CC(C(=O)Nc3nccnc3Cl)C2)c(Cl)c[nH]c2nccc1-2 CC(C)C(F)(F)CC(=O)N1CCC(C(C)NC(c2c(Cl)nsc2Cl)=O)CC1 N1(C(=O)CCc2csnn2)CC(C(N2CCC(O)(C(F)F)C2)=O)C2(CC2)C1 CC(C)(C)C(CNC(=O)COC1CC=CC1)NC(c1ccc(Cl)nc1)=O N1(C(CC(C)(F)F)=O)CCCCC(C2CN(C(c3cc(=N)[nH]c(=N)[nH]3)=O)C2)C1 c1(C(C(=O)NC2CC(NC(c3cc(CC)[nH]n3)=O)C(O)C2)O)ccc(Cl)cc1Cl N1(C(CNS(CC)(=O)=O)=O)Cc2ccccc2OC2(C1)CN(C(C1(SC)CC1)=O)C2 c1(C(N(CCNC(c2c(CC)occ2)=O)CC)=O)ccc2cnccc2c1 c1(CC)cc(C(N2CCC(CN(C)C(C3CC4C=CC3C4)=O)CC2)=O)cc(O)n1 C1(C(=O)NC2(CNC(C3(CC)CCCCC3)=O)CCCC2)CC2OC(=O)OC2C1 CC1CC(C(=O)NC2CC2NC(=O)C(F)(F)C(F)F)=NO1 c1(C(=O)NCC2(NC(C3(O)CC4CCC3C4)=O)CCCC2)ccc([N+](=O)[O-])cn1 N1(C(CSCC#C)=O)CCOCC1CNC(c1cnccc1OC)=O N1(C(CN(c2cnn(C)c2)C)=O)CCCCC1Cn1cc(CCC#N)nn1 Cc1n[nH]c2nc(O)c(C(=O)NC3CCC(CSc4ccccc4)CC3)cc12 C(=O)(N=c1cncc(Cl)[nH]1)c1nc(NC(CN(C)C(c2ccccc2)=O)=O)sc1 C(=O)(CCCCCNC(N)=O)NCC(C)NC(C1CC1C)=O C(=O)(C(C)C(C)NC(=O)C(=C1CCCCC1)F)N(C(C(=O)OC)C)C C1(O)(C(C)NC(c2cc(C(CC)C)no2)=O)CCN(C(c2cocc2C)=O)CC1 c1(CN2C(C(=O)Nc3c(Cl)nc(C)c(C)n3)CC3CC32)cc2ccccc2cn1 CCC(O)CC(=O)NC12CC1CN(C(=O)Cc1sc(O)nc1O)C2 CC1(CO)CCCN1C(=O)CCNC(c1cc[nH]c1)=O N1(C(c2c(C)cc(F)nc2)=O)CCC2(CCN(C(=O)CC3CC4CC4C3)CC2)C1 c1(C(=O)OC)ccnc(N2CCN(c3ccc(NS(=O)(=O)CC#N)cn3)CC2)n1 C#CCC(CC(=O)N(C)Cc1cn(C)cn1)NC(=O)CCCN1CCCC1 c1(CN(C(=O)C(=O)NCC2COC(C)(C)O2)CC)ccc(OC)c(OC)c1 C1(NC(CCC(=O)NCC)=O)CCN(C(=O)C(C)n2cnnn2)CC1C C1(NC(C(C)OCC#C)=O)CN(C(=O)CC2CCN(S(C)(=O)=O)CC2)CC1C c1(C(=O)NCC2(F)CN(C(C(C)CC3CCC3)=O)C2)cnc(O)n(C)c1=O c1(NC(CSCC(=O)NCc2nnc(OCC)s2)=O)cnn(C(C)(C)C)c1F n1(C(C)C(=O)NC2CC(CNC(C3CSC3)=O)C2)cnc2ccccc12 N1(C(C2(C=C)CCC2)=O)CCC2(C1)CN(c1nccnc1F)C2 c1(C(N2CCN(C)CC2C(N)=O)=O)cccc(S(C)=O)c1 O=C1CC2CCCC(CN1)N2C(c1cccc(Cl)c1Br)C(=O)NCc1cccs1 c1(C(=O)NCCC2CN(C(CC(CC)C3CCC3)=O)CC2C)ccc(N)c(O)c1 N1(C(C(N)=O)=O)CC2CC1CCC2NC(C1CC2(CCOCC2)C1)=O C1(C(N(C(C#C)C2CCC2)C)=O)(NC(=O)C(C#N)CC)CC(C)(C)C1 C(C)(CO)(C(=O)NCC(C1CC1)NC(=O)CC(C)c1cccnc1)OC c1(C(=O)NC(C(=O)NC2(C(=O)OCC)CC2)C2CCCC2)[nH]ccc1C CC1CCN(C(C2COC(=O)N2)=O)CC1NC(c1ncccc1Br)=O C1(C)(C(=O)NC(C2CCN(C(CC=CC)=O)CC2)C)CCCC(F)(F)C1 c1(C(=O)NC2CC2C(=O)Nc2ccccc2O)cccc([N+](=O)[O-])c1 C1(F)(CNC(c2cc(C)n(C)n2)=O)CCCN(C(=O)CCc2ccccc2)CC1 c1(OCC)cc(Cl)ccc1NC(C1CC(n2cc(COC)nn2)CN1C(C)=O)=O C1(C(=O)NC(C2CC2C(=O)NCCC2CC(C)(C)C2)C)CC2CC(=O)C1O2 c1(C(N2CC(NC(C3CC34CC4)=O)CC3(C2)CC3)=O)cc2cc(F)c(F)cc2[nH]1 N1(C(Cc2c(C)cc(F)cc2)=O)CCCN(C(=O)CCNC(N)=O)CCC1 c12nnc(n1Cc1cccs1)n2Cc1cccs1.Cc1cc(Cn2cccn2)cs1 N1(C(C(C)(C)N2CCOCC2)=O)CC2(CC(NC(=O)CN3CCNC(=O)C3)C2)C1 c1(CCC(=O)NC2CC(O)(CNC(C(C)C3CCCC3)=O)C2)cccc(C#N)c1 N1(C(C2(CC#C)CCCOC2)=O)C2CCC1CN(C(C1(O)CC(C)(C)C1)=O)C2 CC1OC2(C(N3CC(O)(CCNC(=O)Cn4cc([N+](=O)[O-])cn4)C3)=O)CCC1C2 CCC(CC(=O)NCCN(C(c1nc(C(C)C)oc1C)=O)CC1CC1)SC CC(CC(C)N=c1[nH]c2c(F)cc(Cl)cc2s1)NC(=O)CC1(C)CC1 CCC(C(=O)NC(C)(C)C(C)NC(c1ccc(Cl)[nH]1)=O)NC(N)=O C(CCSC)(C(=O)NCCCn1cnnn1)NC(CCCOC)=O C1(C(N2CC(C)C(CNC(C3(C)CC=CCC3)=O)C2)=O)CC2(C1)CC1(CCC1)C2 C=CC1(C(=O)NCC2(C)CCCN(C(=O)C(C)n3cccc3)C2)CCOCC1 CC1CCN(C(=O)C(C)Oc2ccc(C#N)cc2)CCN1C(c1nnn(C)n1)=O C(=O)(C(C)S(C)(=O)=O)N1CC2C(NC(c3c(C)ocn3)=O)(C2)C1 CCS(=O)CC(=O)NCCN(C(c1cn(CC(O)CC)nn1)=O)C1CC1 c1(CC)nn(C)cc1C(=O)NCc1cc(C(=O)NOCC(=O)N(C)C)cs1 C1(C(N2CCN(c3cc(C)[nH]n3)CC2)=O)CCNC12CCCC2 C#CCCCCCC(=O)NC(C)CNC(=O)CNc1ccc(C)cc1 c1(C(C)C)[nH]nc(C(N2CC(CO)(NC(=O)CSc3cccs3)C2)=O)c1[N+](=O)[O-] C1(C(N(CCN(C(C)C)C(c2cnccn2)=O)C)=O)OCCN(C)C1=O CC1CC(NC(=O)C(O)C(F)(F)F)CCN1C(=O)CSc1nc[nH]n1 C#CCC(CC(F)F)NC(=O)C(C)=CCNC(c1ccc(CO)cn1)=O C1(OC)CC(CNC(c2c[nH]cc2Br)=O)N(C(=O)C=C(C)c2cccs2)C1 N1(C(C(CC)CO)=O)CC(C2CCCN(C(=O)Cn3cncn3)C2)C1 N1(C(CC2(CNC(=O)CCc3cncs3)CC2)=O)CCc2ccc(F)cc21 C12(CNC(C(C=CC)O)=O)CCC(NC(=O)CCOc3ccccc3C)(CO1)C2 N1(C(c2cnc(Cl)s2)C(=O)NCCC)CCOCC1CCc1ccccc1 c1(CC(N2CC(NC(COCCCOC)=O)C(O)C2)=O)ncn2c1CCCC2 c1(OC)cc(F)c(C(=O)NC2CCC(C)N(C(=O)C3=C(C)OCCS3)C2)c(F)c1 CCCC(CC)CCC(=O)NC(c1ccc(CNC(=O)C(C)(CC)CC)cc1)C CCCCC(CNC(c1cc(C)oc1CC)=O)NC(=O)CC1CCC(O)C1 c1(C(=O)NC(CNC(Cc2c(C)ocn2)=O)(C)C)cc(S(=O)(=O)NC(C)C)c[nH]1 C1(CNC(CN(C(C(C)C)=O)C)=O)CN(C(=O)Cc2cccnc2Cl)CCCO1 c1(C(=O)NCC(CC)NC(=O)CC=CCNC(=O)OC(C)(C)C)snnc1C(F)F C1(C2CN(C(c3ccoc3)=O)C2)(NC(CC(C)C2CCCCC2)=O)CC1 CC1CN(C(C2(C(F)(F)F)CC2)=O)CC1(C)CO.c12ccc(o1)CNC2=O c1(CC)nc(C)oc1C(N1CCOCC1CN(C)C(c1nccnc1N)=O)=O c1(CC)cccc2c(C(=O)NCC(C3CCN(C(=O)CC#N)CC3)C)c[nH]c12 C12(NC(c3cc(COC)on3)=O)CCCCCC1N(C(c1ccoc1I)=O)CC2 c1(C(=O)O)ccc(P(C)(C)=O)nc1.c12cccc(c1)C1(CCCC1)C(C)N2 c1(CCN)ccc2nccn2c1.Nc1cc(NC(N2CC(CC=O)C2)=O)nc(O)c1 C1(C)(CNC(c2c(CC)sc(=N)[nH]2)=O)CCN(C(=O)C(C)c2cncs2)CC1 C(=O)(C(N)CS(C)(=O)=O)NC1CC(CC(=O)OC)NC1 c1(-c2cc(NC(CC3(OC)CCC3)=O)sc2)ccc2c(c1)c1ccccc1n2C C1(CNC(CNC(C2CNC(=O)O2)=O)=O)CC2(CCCO2)C1 Cc1nc(NC(c2csc(NC(c3cccc(Br)c3F)=O)n2)=O)c(F)c(Cl)n1 C1(C(C(=O)NC2C(NC(Cc3c(C)scc3)=O)CC2)O)CCCCCCC1 N1(C(c2onc(CC)c2C)=O)CCC(NC(=O)CCCCCF)C(CC)C1 c1(SC)ccc([N+](=O)[O-])cc1C(=O)NCc1cn(CC(C)NC(=O)CC2CC2)nn1 c1(C(=O)NC2C(C)CCN(C(=O)COc3cnn(C)c3)C2)ccc2nncn2c1 c1(C(=O)NCCN(CC(C)O)C(=O)CC2C(C)(C)C2(C)C)ccc2c(n1)NCC2 C1(OCC)CCCC(NC(=O)COCCNC(C2CC2(C)C(F)F)=O)C1 N1(C(CCN2CC(=O)NCC2)=O)CCCC(O)(CCNC(c2ccc(Cl)o2)=O)C1 N1(CC)CCC(NC(C2(NC(C3CCCC(=O)N3)=O)CCOCC2)=O)C(C)C1 C1(NC(c2cc(C)c(C)o2)=O)CC2CC(NC(=O)C(C)(C)COC(C)C)C2C1 CCC(CC(C)C)C(=O)NCC(CC(=O)Nc1cccc(C)c1)OC C=C(C)C1CCC(C)(O)C(NC(=O)CC2CCC3(CCNC3)CC2)C1 c1(C(=O)NC(CNC(C2CCN(CCC)CC2)=O)C(C)C)cc(C)c(C)c(F)c1 N1(C(C(c2cn(C)nn2)NC(C2C(C(=O)OCC)C2)=O)=O)CCC(C)(CO)C1 N1(S(C)(=O)=O)CCN(C(=O)Cc2cscn2)CC1.C12(CCCC1)C(=O)N2C1CC1 C1(C(=O)NCCCOC2CN(c3ncc(F)cn3)C2)CC(=O)NC(=O)C1 c1(C(=O)NC2(C)CC(NC(C3(OC)CC3)=O)C2)nc(C(F)(F)F)n2ccncc12 C(C(=O)NCC(C)N(C)C(C1CC(N(C)C)C1)=O)(C1CCC1)OC C(CN=C(NC(C1CC1)C1CC1)NC1CCCS(=O)(=O)C1)c1onc(C)n1 C1(NC(C(C)=CC)=O)CCCC1NC(c1ccc(CC)[nH]1)=O C(=O)(CC(C)(C)N(C)C(c1cnc(CC)o1)=O)NCc1onc(CC)n1 Cc1cc(CN2CC3C(C(N4CCC(n5cnnc5)CC4)=O)C3C2)cc(C)n1 S(=O)(=O)(c1ccc(N(C)CC2CC2)cc1Cl)NCC1OCC(C)C1 c1(C(=O)NC(CCCCNC(C(COC)(C)C)=O)C)cnn2c1OCC1(CC1)C2 CC#CC1CCN(C(C2CCN(C(C3(C)CC4CCC3O4)=O)C2)=O)CC1 c1(CC2N(C(=O)NCC3CC(OCC)C3)CC2)ccc(F)cc1 C1(C2(O)CCC2)(C(N2C(C(N3CC(OC)C(F)C3)=O)CC2C)=O)CC1 c1(C(N2CCN(C3CN(C(c4c(C)con4)=O)C3)CC2)=O)ccc2nccnc2n1 C1(C)(C(N2CCC(OCC(C)C)CC2)=O)CN(C(C2(C)CCOC2)=O)C(C)(C)C1 C(C)(CO)(C(=O)NC1C(C)CCC1C)NC(Cn1c(C)nnn1)=O Cc1c(C(N2CCN(C)C(CNC(C3CCCCC3)=O)C2)=O)sc(Cl)c1Cl N1(C(c2n[nH]cc2C2CCNCC2)=O)CCCC2(CCCO2)C1 c1(CC)nc(=N)[nH]cc1C(=O)NC1CN(C(=O)CN2CC3CCC2C3)CC1OC C1(C(=O)NCCOCCC)CCN(C(=O)c2ccc(F)c(O)c2)O1 S(=O)(=O)(c1ccccc1OC(F)(F)F)NC(C(=O)OC)(C)C1CC1 C(=O)(C1=C(C)CCOC1)NC(c1ccnn1C)C(N1CCCC(CCC#C)C1)=O C1(NC(c2c(OC)ccs2)=O)CN(C(c2nnn(C(C)C)c2C)=O)CC1OC Cc1c(C(N2CCC(NC(C3CS(=O)C3)=O)C2)=O)cncc1Cl N1(Cc2ccc(NC(C)=O)s2)CC2CCN(C(=O)Cc3noc(C(C)C)n3)C2C1 Cc1ccc(N)cc1C(=O)NCc1csc(CNC(=O)C(C)(C)F)n1 C1(CNC(C(CSC)OC)=O)(NC(c2cc(=O)cc[nH]2)=O)CCCCC1 c1(C(C(=O)NC2CCCCC2)N(C(CCCC)C)C)ccc(F)cc1C c1(C(N2C(CCNC(C3(CCC)CCOC3)=O)CCC2)=O)nc(C(C)C)oc1C c1(C(=O)NCCc2n(C(C)C)c(S)nn2)c[nH]c2nc(Br)ccc12 C(C)(N=c1nc(N2CC(F)C(F)C2)c2sccc2[nH]1)c1c(NC(C)=O)cccc1 CCC(C(=O)NCCNC(=O)Cc1ccno1)C1CCOCC1 Nc1ncccc1CC(=O)NCC1CCN1C(=O)COc1ccc(Br)cn1 Cc1nc(C(=O)NC2CC(NC(c3csc(C4CC4)n3)=O)C2)c2ccnc-2[nH]1 Cc1cc(=NC2CC3C(C2)C3(F)F)[nH]c(=NCC(=O)NC(C)C)[nH]1 CC1(NC(=O)CSc2ccncc2)CCN(C(=O)CC2(C)CC2(F)Cl)CC1 CN(S(=O)(=O)N1CCCC(O)C1)CCC1CCOC1 N1(C(C2(c3cccs3)CC(=O)C2)=O)CC2CC(NC(C3SCCCS3)=O)CC2C1 N1(C(CCN(C)CC)=O)CC2(CCC(NC(c3ccc(NC)c(F)c3)=O)CC2)C1 C(C1CN(C(=O)C(C)CC(N)=O)Cc2ccccc21)NC(CC(CCC)O)=O c1(CN2CCC(CS(=O)(=O)NCC(F)F)CC2)ccc(F)c(C(F)(F)F)c1 C(C)(CN=c1[nH]c2c(c(=NC(C)c3nc(C)cs3)[nH]1)CCC2)n1c(C)cc(C)n1 N1(C(N2c3ccc(C(C)(C)C)cc3CC2)=O)CC(=O)CC(P(C)(C)=O)C1 C(=O)(C(F)CC(C)(C)C)N(CCN(C(CCN(C)CCO)=O)C)C c1(C(=O)NC2C(NC(CCCC)=O)COC2)cccc(OCc2cnn(C)c2)c1 C1(C(C)C)COCCN1C(=O)CC1CCCCC1NC(C1(N(C)C)CC1)=O C1(C(C(=O)NCC(=C)C)N(CCCO)C)CC2CCC1O2 CC(C)CC(O)CC(=O)NC1CCC1C(=O)NCCC(=O)NO Cc1cc(C(=O)NCC23CC(NC(c4ccc(CO)s4)=O)(C2)C(C)O3)cc(Cl)c1 n1(CC(=O)OC)nc(C)c2ccc(C(NC3c4ccccc4CC3O)=O)cc12 C=CC(C)CC(=O)N1CCCC(NC(c2cc(Cl)cn2CC)=O)C1 C#CCC(C(=O)N(C(=O)CCC(C)=O)C(c1ccc(F)cc1)CC)C1CC1 c1(C(=O)OCC)cc(N2CC(F)CC2CNC(c2c[nH]nc2C)=O)nc(C)n1 n1(C(C)C)ncc(F)c1C(=O)NCCNC(=O)C(Cc1ccsc1)NC=O c1(OC)ncnc(OC)c1C(=O)NCC12CCC1CN(C(C1CCO1)=O)C2 c1(C(=O)NCCOCCNC(C(CSC)C)=O)cc2cc(C)c(C)cc2o1 C=C(C)C(O)CC(=O)NCCCCCNC(=O)Cc1c(C)noc1Cl CCS(=O)(=O)CC(=O)N(CC(=O)NCc1cnc(C)s1)C C1(N(C)C(C2CCCCO2)=O)CCCN(C(c2ccc(N)c(C(F)(F)F)n2)=O)CC1 Cc1ccc(Cl)c(OC(C)C(=O)NC2CCOC(c3cnn(C)c3)C2)c1 C(=O)(C(Cc1ccccc1)C(C)C)N1C(C(C)NC(CCC(=C)Cl)=O)CCC1 CCC(O)C(C)C(=O)NCc1ccc(C(=O)NOCc2ccc(C)cn2)s1 C1(C(N(C(CNC(c2c(C)noc2C(F)(F)F)=O)C)C)=O)CCc2nncn2C1 c1(C(N2CCN(c3ncc(C)cn3)C(C(C)C)C2)=O)cc(Cl)cc(Br)c1Cl C1(NC(C(c2c(C)noc2C)C)=O)CC2(CCN(C(C3CC3C#N)=O)C2)C1 CC(CC(=O)NCC(C1CCCC1)NC(=O)C(C)(C)c1cccs1)NC(N)=O C1(CNC(CN(CCC)C)=O)(NC(c2cnc[nH]2)=O)CCC(C)(C)CC1 C1(C(N(C)Cc2[nH]ccc2CNC(=O)CC2CSCCO2)=O)CCCCN1C CCC(C(=O)NC(C1CCCN1c1nnc(CO)s1)(C)C)n1cccn1 C1(C(N(C2CCCN(C(=O)CC=C(Cl)Cl)C2)CC)=O)CCC2CC1CO2 C1(CCCNC(=O)Cn2nnnc2C2CC2)CN(C(C2CC3CC3C2)=O)CCO1 C1(NC(c2cc(CC(C)C)on2)=O)CCN(C(=O)COCC(F)(F)F)C1C C(CNC(=O)CC1CC(NC(C2CCC(=O)NC2)=O)C1)(C(C)(C)C)OC C1(CNC(CCC(=C)Cl)=O)CCN(C(c2cc(C(C)=O)c[nH]2)=O)CC1(F)F C1(C(=O)NCCNC(c2cc(COC)no2)=O)CC12CC(C)(C)C2 C(C)(C(=O)NCC1CC2(CC2)C(=O)O1)(C(C)C)NC(C1CC(COC)C1)=O C1(C(=O)NCC2(C(=O)NCc3ccccc3)CC2)CCCOCC1 N1(C(c2c(C)ccs2)=O)CC(C2(NC(=O)C(C)NC(C3CCCC3)=O)CC2)C1 c1(CC)cncc(CNC(=O)C(C)N(C(=O)C(C)OC2CCCC2)CC)c1 C(=O)(C#CC1CCOCC1)N1CC(C)(OCC(=O)NCCC(COC)O)C1 c1(C(C)=O)ccc(-c2cn(-c3ccc(C(=O)NC(C)CN(C)C)cc3)nn2)cc1 Cn1cnc(CCC(=O)NC(C)(C)C=CC(N2CCC(N3CCCC3)C2)=O)c1 c1(C(=O)NCCC2(O)CN(C(c3n(CC)ncc3Cl)=O)C2)c(C)ccc(C)c1O C(=O)(C(CCc1ccccn1)N1CCCC(CN(C)C)C1)NCCCC CC1=C(C)CC(CNC(c2cncc(F)c2)c2nnnn2-c2ccccc2)CC1 Cc1ccc(CC(N2CCC(N(C(=O)C(C3CCCCC3)F)C)C2)=O)cc1O c1(C(N2C(CNC(CC3CCC(C)CO3)=O)CC2)=O)cnc2ccccc2n1 C(=O)(C(CO)C(C)(C)C)NC(CC(C)C)C(=O)N1CCC(CNC(C)=O)C1 c1(C(N2CCC(C)(C)C(NC(c3cnc(O)o3)=O)C2)=O)ccc2cccnc2c1 c1(NC(C2(C)CN(C(c3ccc(F)c(Br)c3)=O)C2)=O)cccn2ccnc12 C=CC1CN(C(=O)C(CC2CCOCC2)NC(=O)CC2COCCO2)CCO1 CCCC(C)(C)C(=O)N1CCC1C(N1CCOC(C(C)C)C1)=O Clc1nc(I)ccc1CNc1ccc(-n2ccnn2)cc1 CC(C)CC(CNC(C1CCC(N(C)C)CC1)=O)NC(c1ccc(CF)cc1)=O C(CCCC(C)NC(c1c[nH]c(=O)cn1)=O)NC(C(CC)N(C)C)=O c1(OC)cc(F)c(CC(=O)NCC(CO)NC(=O)C(c2cncnc2)C)c(Cl)c1 C(CCC)(C(=O)NC1CCC1CNC(C1(c2cccc(F)c2)CC1)=O)=CCC n1(CCCSCC)c(N(C)CCOC(C)CN(C)C)nnc1-c1ccco1 C1(NC(C2CC(C)(C)C2)=O)CCCCN(C(C2CC2c2ccc(F)cc2)=O)C1 c1(C2C(F)(C(=O)NCC(C)N(C)C(C3CC3)=O)C2)ccccc1.c1ccccc1 c1(C(N2CCCC(NC(CC3CC(=C)C3)=O)C2C)=O)nc2ccccc2n1CC c1(C(N2CC=CC(NC(C3ON=C(CC)C3)=O)C2)=O)cc2cccnc2[nH]1 C1(NC(=O)COc2ccccc2F)CC2CN(C(=O)Cn3cccn3)CC2C1 N1(C(CCCC)=O)CC(C2CC2C(=O)NCC2(O)CN(C)C2)C1 C(C(COC)C(=O)NCC1(CNC(=O)Cn2cnnc2O)CCCC1)OC C(=O)(C(C(C)(C)C)NC(N)=O)NC(CC(C)NC(C1CCOC1)=O)C c1(C(=O)NC(COCC)C(=O)NC(C(F)(F)F)C2CC2)ccc(C)nn1 C=C(C)CC(C)C(=O)NCC1COCC1NC(c1ccc(OC)c(OC)c1)=O N1(C(c2c(CC)cco2)=O)CCN(C(=O)C=CC(C)CC)C2CC12 c1(OC)ncc(Br)c(=NCC2(F)CC(NC(c3ccccc3SC(F)F)=O)C2)[nH]1 c1(OC)cc(CC(N2CCC(C)(NC(=O)Cc3nc(=N)[nH][nH]3)C2)=O)cc(F)c1 C1(NC(C(CC#C)O)=O)CC2CCC1N2C(C1CC2C=CC1C2)=O C(=O)(C(CC(C)(C)C)NC(C1CC2(CCC2)C1)=O)N(C)CCOC(F)F N#Cc1sccc1C(=O)Nc1cccc(NC(=O)CCCC2CCCO2)c1 CCC(C)(C)C(=O)C(=O)NC(CC1CC1)C(=O)NC(C1CCCC1)CO C(=O)(C1=CCCOC1)N(C)CC1CC(F)CN1C(C1CCS(=O)CC1)=O C1(CNC(CCCN(C)N=O)=O)CN(C(C2CC=CCO2)=O)CC2(CCC2)O1 C=CCC(C(=O)N(C)CC1CCCCN1C(=O)CC(OCC)OCC)N(C)C C1(N(C(c2cc(F)ncc2Br)C(=O)NCC=C)C)CC(C)OC(C)C1 CN1CCC(NC(c2cc(CNC(c3ccn(C4CC4)n3)=O)[nH]n2)=O)C1 Cc1cc(Cl)nc(N)c1C(=O)NC(c1ccc(CNC(C2CCCS2)=O)cc1)C C(=O)(C(C)(O)CC(F)F)NCC1(C)CCN(C(C(=O)NCC)=O)C1 C(CC(CC)C(=O)NC(CCN(C)C(C1CC(F)C1)=O)C(C)C)=CC C1(NC(C(C=C=C)C)=O)CC2CC(NC(=O)Cc3cccc(Cl)c3)C2C1 C(CCC1CC1)(C(=O)NC1(C2CC2)CC1)NC(c1cc(COC)[nH]n1)=O N1(C(c2cn(CCC)nn2)=O)CC(NC(=O)C=Cc2cnn(C)c2)CC(C)C1 C1(CNC(CNC(=O)NC)=O)C(C)CCCN1C(=O)CC1(O)CCCCC1 C1(C(=O)NCC(CNC(c2c(CC)occ2)=O)O)Cc2nncn2C1 C(CC(C)C)(C(=O)N1CCC1C1CCOCC1)NC(c1[nH]cc(C)c1)=O N1(C(C2(NC(=O)Cc3csnn3)C(C)(C)C2)=O)CCC(C2CCCC2)C1 C12(C(=O)NC(CC=C)CC=C)CCN(C(c3cc[n+]([O-])cc3)=O)CCC1C2 CC(CN=C(NCCOc1ccc(Cl)c(F)c1)NC1CCCC1)N1CCN(C)CC1 C12CN(C(C)(C)C1)C(=O)C(C)N(C)C1(CC1)C(=O)N2.c1(SC)ccccc1 C12CC3CCCCC3N1C2.c1(C(=O)NCc2n(C)nnc2)n[nH]c2c1CCC2(F)F C1(C(=O)NCCC2CC2)CN(Cn2c(O)nnc2O)CC12CC2 C1(C2CCCOC2)(NC(=O)Nc2ccc(F)cc2Cl)CC1 n1(CC)nc(C(=O)N(C)CC2CCCN2C(c2ccc(OC)cc2)=O)ccc1=O C1(NC(C2(COCC)CC2)=O)CCCCN(CC(n2cc(COC)nn2)C)C1 C1(SCC(=O)NCc2nc[nH]n2)CCCCC1C(=O)NCCCCn1ccnc1 C1(CNC(CCC#C)=O)C(O)C(O)CN1C(C1CC(C(F)F)(OC)C1)=O CCCCCC(CNC(c1cc(Cl)ccn1)c1nnnn1CCSC)CO C1(C#N)(C(=O)NCCCNC(c2nc(C(C)OCC)sc2)=O)CC12CCC2 C=C(C)CC(C(=O)NCc1ccn(C)c(=O)c1)NC(=O)C(C)CC=CC c1(C(N(C2CCN(C(c3c(C)nn[nH]3)=O)C2)C)=O)ccc(I)c(Cl)c1 CCC(C(=O)N(C1CN(C(=O)C=Cc2cocn2)CCC1O)C)C(C)C c1(C(N2C(CC(=O)NCc3ccc(Cl)s3)CCC2)=O)ccc(O)c(Cl)c1 C(=O)(C(C)C(C)(F)F)NC1CN(C(c2cc(C(C)C)oc2C(C)C)=O)C1 c1(OC)cccc(SCC(N2CCC(C)(NC(=O)CCNCC(F)(F)F)C2)=O)c1 C1(NC(CC2(O)CCN(C)CC2)=O)CCC(N=c2[nH]c(Cl)nc3[nH]cnc23)CC1 N1(C(C2(C)C(C)CN(C(C3COCC(C)O3)=O)C2)=O)CCC2(CCC2)CC1 C1(CC(=O)NCC(C)N(C(=O)COCCOCCO)CC)CCCCCCC1 C1(CC)(NC(=O)Cc2cc(OC)ccc2F)CCN(C(C2COC(C)C2)=O)CC1 c1(C(c2n(C(C)C)nnn2)NC2CC2c2ccccc2F)c(Cl)nc(Cl)n1C S(=O)(=O)(c1ccccc1[N+](=O)[O-])NCC(N1CC=CC(NC(CN(C)C)=O)C1)=O c1(N(C2CN(C(=O)C(CC)n3cccn3)C2)C)nc(O)c2cnn(C)c2n1 c1(-c2ccc(C34SCC(C(=O)O)N3C(=O)CC4)cc2)ccc2c(O)nccc2c1 c1(CC(=O)NC(CNC(C2(C=C)CCC2)=O)C(C)C(C)C)cnc2n1CCOC2 c1(C(=O)NCC2CCC(NC(C3(C=C)CCC3)=O)C2)sc2cccnc2c1Cl N1(C(C=C(C)C(F)F)=O)CCC(CO)(NC(C2CC(C)(C)C2C(F)(F)F)=O)CC1 C1(COC)(NC(c2cnn(C(C)C)n2)=O)CCCN(C(c2cnccc2C)=O)C1 C1(C(N(CC(=O)NC2CCCC(CO)CC2)C2CCC2)=O)CCC2(CC2)CO1 c1(OC)ncc(NC(C2CCCC2NC(c2ncccc2Br)=O)=O)cc1Br c1(C(C)Nc2cc(NCc3cccc(SCC)c3)ncn2)ccc(Cl)cc1Cl C(=O)(CCCCC#N)N1CCC(CCC(=O)N(CC(=O)NC(C)(C)C)C)CC1 c1(OC)cc(C(=O)NCC2C=CCN2C(c2cnc(Cl)[nH]2)=O)cc(Cl)n1 C1(C(=O)NC2CC(OCC(=O)NCCSC)C2)CCOC1C1CCC1 c1(C(=O)NC2CC3CC(NC(CN(C)C(N)=O)=O)C3C2)noc2cc(F)ccc12 CCC(CC)CC(=O)N(C1CC(NC(C2(CC)CC2(F)F)=O)C1)C CC1CC(NC(=O)CCn2cncn2)CCN1C(C1CC12CC(C)(C)C2)=O c1(CCc2cn(C3CC(NC(C(C#N)C4CC4)=O)C3)nn2)cc(Cl)sc1Cl Cc1cc(O)ccc1C(=O)NC1CC1NC(=O)C(C)Cn1ccnc1 c1(C(N2C(CNC(COC(C)C)=O)CC3COCC32)=O)c2c(c[nH]c1=N)CCC2 C=CCC(C(=O)NC1(C(=O)NC(C2CC2)C2CC2)CC(O)C1)C(C)C Cc1nnc(CCC(=O)NCC2(C)CC(NC(=O)CN3CCCC3C)C2)n1C C1(NC(c2ccc(C)nn2)=O)CCCCCC1C(=O)NC(C)C(C)C C1(NC(CC2(C=C)CCC2)=O)CCCN(C(=O)C=Cc2nc(C)co2)C1 CC(F)CC(=O)N(C1CCN(C(=O)Cn2cc(Cl)cn2)C1)C Cc1cc(C#N)sc1C(=O)NC1CCN(C(c2ccn(CC(C)C)n2)=O)C1C c1(CC(=O)NC2CC2NC(C2CC3C=CC2C32CC2)=O)ccc2n[nH]cc2c1 C(=O)(CCCC(C)NC(c1ncn2c1CCC2)=O)N(C(C)CC1CC1)C C1(OC)CC(CNC(c2csc(=N)[nH]2)=O)N(C(=O)C(C)C2CC2)C1 c1(OCC#C)cc(OC)cc(-c2cn(CCC3CC34CCCC4)nn2)c1 C=C(Br)CC(C)(C)C(=O)NC1CN(C(c2cnn(C)c2C)=O)CC1C(F)F c1(CC(N2C(CCCNC(C3CCCC3CF)=O)CCC2)=O)sc(O)nc1O C(=O)(C1=CCCCC1)NCC(CC=C)NC(c1cccc(Cl)c1C)=O c1(-c2cccc(OC)n2)ccc2c(C(=O)Nc3cnnn3C)nn(C)c2c1 Cc1ccc(C(O)CSCC2CCCOC2)cc1 c1(C(=O)NC(CC=C)CNC(=O)CSc2ccc(C#N)cc2)noc2c1COCC2 Nc1cc(F)c(C(=O)NC23CC2CN(C(c2ccc4ncccn24)=O)C3)c(F)c1 CN1N=C(C(=O)N2CCN(C(c3c(O)cccc3O)=O)CC23CC3)CCC1=O N1(C(c2ccc(-c3ccc(C(C)=O)cc3)o2)=O)CCN(c2nncs2)CC(O)C1 N1(C(c2cc(C#N)on2)=O)CCC(C2CN(C(c3cc(CO)on3)=O)C2)CC1 Cc1cccc(C)c1CN(C(=O)CCCc1nnc(-c2ccc(Cl)cc2)o1)C c1(C(=O)NC2CN(C3CN(C(c4cccs4)=O)C3)C(=O)C2)c[nH]c2cccnc12 C(CCCCCC(=O)NC1(CF)CCC1)n1cc(C2C(C)NC(=O)CC2)nn1 C12(CNC(CC=CCC)=O)CCC1CCN2C(c1n[nH]c(CC)c1Cl)=O C12(CNC(c3nc(C(C)(C)C)[nH]n3)=O)CCCC1CCN2C(C1CCCC1)=O N1(C(C(C)N(CC)CC)=O)CCC(CO)(CNC(=O)CCC2CC2(Cl)Cl)CC1 N1(C(c2cc(C(=O)OC)on2)=O)CCCCC(N(C)C(c2c(C)n[nH]c2C)=O)C1 N1(C(C2(C)CCN(C(C)=O)C2)=O)Cc2ccc(Cl)cc2C(C)C1 C1(C(=O)NCCC2N(C(CC3(N(C)C)CCC3)=O)CCC2)CCC2(CCC2)CC1 C1(C)(CC(=O)NC(C)CCNC(=O)CC(F)(F)F)CCS(=O)(=O)N1 N1(C(c2ccc(C(=O)OC)s2)=O)CCC(NC(c2cc(C)co2)=O)C(C)C1 N1(C(CCOC)C)CCn2c(C(F)F)nnc2C1 c1(N(C(CN(C(CC)C)C)=O)C(=O)Cc2cccc(O)c2)ccccc1OC C=CC(C)C(C)C(=O)NCC1(CO)CCN(C(C2(C3CCC3)CC2)=O)CC1 c1(C(N(C2CC(NC(CCC(C)C)=O)C2)C)=O)cc2ccncc2cc1F c1(COC)cc(C(=O)NCC(C)(O)CNC(=O)C(C2CCOCC2)OC)cs1 C1(C(=O)NC(CC#CC)C)C(C2CC2)CCN1C(C1CCCCC(=O)N1)=O N1(C(CCCC)=O)CCC2CCCC12CNC(c1cccnc1-n1ccnc1)=O N1(C(C2(C)CC2)=O)CCCC(C2CN(C(C3OCCC3(C)C)=O)C2)C1 C1(C(=O)NC(CO)C(C)NC(C2CC3C(C2)C3(F)F)=O)(OC)CCCCCC1 N1(C(C2CN(C(CCC(=C)Cl)=O)CC2(F)F)=O)CCC2CC1C(=O)O2 C1(NC(C2(C(N)=O)CC2)=O)CC2CCC1N2C(=O)CN1CSCCSC1 c1(-n2cc(C3N(C(CC4CCC(OC)CC4)=O)CCC3)nn2)cccc(F)c1F O=C1CCC(C(=O)NCC2(CO)CCN(C(=O)CCc3cnc[nH]3)C2)CCO1 C1(NC(c2ccc(NC(C3CC34CC4)=O)o2)=O)(CSC(F)F)CC2CCC1CC2 C=C1CCC(C(=O)N(C)CC=CC(=O)NC(CO)C2CCC2)CC1 CCC(CN(C)C)CC(=O)N1CC(O)CC1CNC(=O)CCn1ccc(C)n1 CCCC(C)(C)CC(=O)NC1CCC(C)(CNC(C2(CC(=O)OC)CC2)=O)CC1 C(=O)(CC(C1CC1)NC(C1CC(C)N1C(=O)COCCCF)=O)NC C(C(CO)N=c1[nH]c(Cl)nc2c1CCC2)NC(C(C)(C)O)=O N1(C(COC(CC)C)=O)CCN(C(=O)COC2CCC2)CC1CCO C(=O)(CC(C(F)F)n1cccn1)N(C1CCCN(C(=O)Cc2ccc(O)cc2)C1)C C(=O)(CCCC(F)(F)F)NCC(C)C(F)C(=O)NC1CCCCC12CCC2 C1(CNC(CC2C(C)(C)CC2)=O)(NC(c2ccc([N+](=O)[O-])o2)=O)CCCCCC1 c1(C(N2C(C)CCN(c3ccc(F)cn3)CC2)=O)ccc2ccn(C)c2c1 C(=O)(CCC(CC)NC(=O)Cc1cccnc1)N(CCCC)CC(N)=O C(=O)(CC(C(F)(F)F)P(C)(C)=O)NCC1CCN(C(C2(C)CCOC2)=O)CC1 N1(C(CCCCC#C)=O)CC2CC(C)N(C(=O)Cc3cc(CC)nn3C)C2C1 C12(CNC(c3ncc(C)nc3)=O)CN(C(=O)CC3CCCC(=O)C3)CC1CCO2 CC1(C)C2CCC1(C)CN(S(=O)(=O)c1ccc(NCC=CCl)nc1)C2 N1(C(c2cccc(C)c2)=O)CC(NC(=O)CC2CCC3(CCC3)O2)CC(O)C1 N1(C(C=CC=CCC)=O)CCC2CCN(C(=O)Cc3c[nH]ccc3=O)CC2C1 C(=O)(C1=CCCCCC1)N1C(C)CC(NC(c2ccc(-c3ncon3)cc2)=O)C1 c1(SCC2N(C(=O)NC3CC(n4cccn4)C3)CCC2)ccccn1 O=C(O)CC(CN1CCOCC1)NC(c1sncc1C(F)(F)F)=O N1(C(CCCNC(C)=O)=O)CCCC(CCNC(C2CCCC3(CC3)C2)=O)CC1 C#Cc1cc(C(N2CCC(NC(C3CCCN3C(C)=O)=O)C2)=O)cc(Br)c1 Cc1ccnc(C)c1NC(C1CCCCN1C(=O)CCc1cnoc1)=O C(=O)(C(CC(=O)NCC(O)CC(F)(F)F)NC(=O)OCc1ccccc1)OC N1(C(CCC(=C)Br)=O)CC(NC(=O)C(=Cc2cccnc2)F)C2CCCC2C1 c1(C(=O)NCC(CC)(C)NC(C2CCSCC2)=O)cnc2ncnc(O)c2c1 c1(NC(CCC)CCCC)ncccc1S(=O)(=O)NCC(C)(C)C(C)C N1(C(C(=O)NCC)=O)CC2CC1CCC2NC(C12CCCCC(OC)(C1)C2)=O c1(C(C(=O)NCCOC)N(C(CC)COC)C)ccc2c(c1)CCCO2 C1(CC(=O)NCC(CC(C)C)NC(C(=O)NCC)=O)CC(=O)c2ccccc2C1 Cc1nn2cc(C(N3CC(CO)(NC(=O)Cc4cc(O)nnc4O)C3)=O)nc2s1 N1(C(C(CC=C)C(C)C)=O)CC(NC(=O)CC2=CCCC2)C(S(C)(=O)=O)C1 C1(C(=O)NC2CC(NC(c3cccc4cc[nH]c34)=O)C2)CC2CCC(C1)S2(=O)=O c1(C(=O)NC(C(=O)OC)Cc2cn(CC(N)=O)nn2)cncc(Cl)c1 Nc1c(O)ccc(Cl)c1C(=O)NCC1CC12CCN(C(C1CCC(=O)N1)=O)CC2 c1(CN2CCC3CN(C(C4=C(C)OCC4)=O)CC3C2)cccc2c(Br)ccnc12 Cc1cc2ccccc2n1CC(=O)NCCN(C(=O)C(CO)C(C)(C)C)C(C)C c1(CN2CCCC(C(=O)Nc3ccc(CC)cc3)C2)cc(Cl)c(O)cc1O CCCC(CC)C(=O)N1CCC(CNC(=O)C(=O)NCC2CC2)C1(C)C CC(=NO)c1sc(NC(c2cccc(C3CCOC3)c2)=O)nc1C N1(C(C(C)C#N)=O)C2CCCC1CN(C(C1CCCCC1C(N)=O)=O)C2 c1(C(=O)NC(C)C(CO)NC(=O)C(O)C(C)(C)C)cccc2c1CCC2 CC1CC(C(=O)NCCC2COC(C)(C)C2)CN(C(=O)Cc2ccnn2C)C1 N1(C(CC(CC(=O)OC)C)=O)CCC2OCCN(C(C3CCC(C)CC3)=O)C2C1 c1(C(=O)OC)ccc(F)c(C(=O)NCC(C)N(C)C(C2CNC(=O)N2)=O)c1C N1(C(CC(C)NC(CCN(CCC)C(C)=O)=O)=O)CCN(CCO)C(C)C1 C1(N(C)C(c2ccco2)=O)CCCN(C(C2(c3ccccc3)CNC(=O)C2)=O)C1 C(CNC(c1cc(Cl)ns1)=O)(CC(F)(F)F)NC(C(C)SC)=O c1(NC(C(C(C)SC)O)=O)nc(C)cc(C#N)n1 C1(NC(C(C)(C)N(C)C)=O)CCN(c2ncnc3c2COC3)CC(C)(C)C1 N1(C(CCC(=O)NCC)=O)CCN(C(=O)CC(F)(F)CC)CC1c1ncc[nH]1 c1(CNC(=O)Nc2ccc(C3CCC3=O)cc2)cc(F)c(F)cc1Cl Cc1cc(C)c(C(=O)NC2(C3CCCN3C(=O)CC3COC(=O)C3)CC2)o1 N#Cc1cc(Cl)c(C(N2CC3(NC(=O)CSCc4ccncc4)CC2C3)=O)s1 c1(C(=O)NCC=CCNC(Cc2cc(C)sc2)=O)cccc2ncc(C)n12 C1(C(=O)NCCOCCCNC(C2CCN(C(C)=O)C2)=O)CCCC(=O)O1 c1(NC2(CNC(c3cccs3)=O)CC2)ncnc2c1CCC2 C1(C(=O)NCc2ccc(C)c(C)n2)CCN(C(=O)OC(C)(C)C)C12CCC2 CON1CCC(C(N2CCCC(C)(NC(=O)Cc3ccc(F)cn3)C2)=O)CC1 CC#CCC(C(=O)NOCCC)NC(C1CC1C1CCC1)=O N1(C(c2ccnn2CCF)C(=O)NC)CCC2(CCCC2CN=[N+]=[N-])CC1 C(C)(CS(=O)CC)NCc1ncc(COCC)[nH]1 C(=O)(CCCC(C)C)N1CC(NC(C2(C(=O)OC)CC2)=O)C(n2ccnn2)C1 C1(N(C(c2cc(CC)[nH]n2)=O)C)CCN(C(=O)CNC(=O)OC)CC1C Cc1csc2ccc(C(=O)NCCCN(C)C(C3C(C)OC(C)C3C)=O)cc12 Fc1cccc(CNN2CCN(c3ncccn3)C(CC3CC3)C2)c1C C(CC(CNC(=O)C(C)(C)C)NC(c1cnc(-c2ccsc2)s1)=O)OC N12CC(C3(CC3)C1)C2=O.Cc1ccnnc1NC(=O)C(C)Oc1ccccc1Cl C1(N(C)C(C2(C3CCCO3)CC2)=O)CCC(NC(=O)C=C2CC2)CC1 Cc1cnn(C)c1CC(=O)NCC1(F)CCN(C(=O)C(=O)NC2CC2)C1 c1(CC(OCC)OCC(=O)OC)nc(Nc2ncccn2)cc(Cl)n1 c1(SC)cc(C)c(C(N2CCCC2c2csc(Br)c2)=O)s1 c1(C(N(CCOCCNC(c2c(C)noc2)=O)C)=O)cnn2c(Cl)cccc12 C(=O)(CCC(C)(C)F)N1C(C(C)NC(c2ccco2)=O)CCC1 C#Cc1ccc(C)c(NC(N2CCC(Oc3ccccc3I)CC2)=O)c1 CC(CC(F)F)C(=O)N1CC2CC2(NC(=O)Cn2cc(Br)cn2)C1 C1(NC(C2(C#C)CN(C(c3ccn(C)n3)=O)C2)=O)CCCCC1(C)C c1(C(N2C(COC)(CNC(=O)C=CC(=O)N(C)C)CCC2)=O)nccn2ccnc12 N1(C(C(C2CCCCC2)C)=O)CC(C(=O)NCc2cnn(C)c2)CC(O)C1 c1(OC)cc(C=CC(N2CC(NC(c3ccncc3Cl)=O)CC2C)=O)ccc1O C1(NC(C2C(OCC)C2)=O)CCN(C(=O)CN2CCC(N(C)C)CC2)CC1F.NCC CC(CCNC(=O)CNC(c1ccsc1)=O)CCNC(C1CCC(C)(C)C1)=O c1(C(N2CCN(C(=O)CC3CSC3)CC(CO)C2)=O)ccn2c(O)nnc2c1 N1(Cc2ccc(OC)o2)CC2(CC(C(=O)NCc3cncc(Br)c3)C2)C1 CC1(NC(C2CCN2C(=O)C(O)C2CCC2)=O)CC=CCC1 c1(-n2ccc(C(=O)NC(CCCC)CNC(=O)CC(F)F)n2)c(C)nn(C)c1C CC(CC(=O)NCC1(CC(=O)NOCC(N)=O)CC1)C(F)(F)F C(=O)(C1=CC2CC(C1)CC2O)N1CCC(C(C)NC(=O)CSc2n[nH]c(O)n2)C1 C1(C(N(C(C(C)C)CO)C)=O)CC2CC1CN(C(c1cc(F)n(C)n1)=O)C2 c1(C(=O)NC2C3CC(NC(C(CC#C)O)=O)CC32)c[nH]c2ccccc2c1=O C(=O)(C(CC(C)(C)C)OC)NCC(c1ccccc1CC)NC(CSCC=C)=O Cc1c(NC(=O)N(C2CCC(=O)NC2)CC2CCC2)cnn1-c1ccccc1F C(=O)(CC(C)N(C)C(c1cc(C)ns1)=O)N(C1CC(OCC)C1)C Cc1cc(N2CC(C(N)=O)OC(C)C2)nc(C2CCC2)n1 CCCC(C)C(=O)NCC(C)(CO)NC(=O)CCc1ncc[nH]1 N1(C(CCC(C)C)=O)CC(NC(=O)C(O)C2=CCCCC2)CC12CCOCC2 CC1CC(NC(=O)C(F)n2ccnc2)CCN1C(c1ccc(-c2ccco2)s1)=O c1(-c2cnc(CN(C)C)s2)nc(-c2ccsc2)nn1Cc1ccccn1 C1(CNC(CC2(C)CCN(C(CC=C(C)C)=O)C2)=O)CC(=O)N(C)C1=O CCC(C)(COC)C(=O)N1CCCC1CNC(=O)Cc1cccc(C(C)C)c1 N1(C(C2OCCC(NC(c3ccn(CCC)n3)=O)C2)=O)CC2OCCN(C)C2C1 C1(NC(c2csc(O)n2)=O)CC12CCN(C(=O)CC1CC(C(F)F)C1)CC2 C1(C(=O)NCCOCCC(C)C)CCC(C2CC2)N1C(=O)Cc1ccoc1 c1(OC)noc(C2CC2)c1C(=O)NC1COCC1NC(=O)CCc1ccco1 C1(CNC(C(CC)C2CCC(=O)N2)=O)C(C)CCCN1C(=O)CC1CCC(C)C1 c1(-c2cn(CC3CN(C(c4c(C)nsc4N)=O)C3)nn2)ccc2occc(=O)c2c1 N1(C(C2N(C(C)=O)CSC2)=O)CCN(C(C2C3CC3C3CC23)=O)CC1C c1(CC(=O)NC(C)C(CO)NC(=O)C(F)C(F)(F)F)cc(F)c(F)cc1F CC(C(C)(C)NC(=O)OC(C)(C)C)NC(=O)NCC1C(C)C1(F)F C1(NC(=O)NC(C2CCCCO2)C)CCOCC12CCCC2 C1(NC(C(C)CC(F)F)=O)CCC2(CC1)CN(C(C1CCCOCC1)=O)CCO2 c1(CC)cc(C(=O)NCCN2CCC(NC(C3(C)CC(C#N)C3)=O)CC2)sc1C N1(C(CCC=CCC=C)=O)CCCCC1C(C)NC(=O)CN1CC2CC2C1 c1(SC)cc(C(N2CC3CC2C3CNC(c2sc(C)nc2C)=O)=O)nn1C C1(NC(=O)Cc2ccc(O)nc2)CN(C(=O)C#CC2CCC2)C2(CCCOC2)C1 Cc1ccc(C)c(C(C)NC2(C(=O)O)CCSCC2)c1 N1(C(C2C3N(C(CN(C)C(N)=O)=O)C(CC3)C2)=O)CCc2sccc2C1 CCC(C)C(C)C(=O)N1CC2CC1(CNC(=O)C(O)C(C)C)C2 N1(C(Cn2cccc(C)c2=O)=O)CCC2CC2(NC(=O)Cn2ccnc2C)CC1 N1(C(c2ccc(C)c(F)n2)=O)CCCN(C(C2CC2F)=O)CC1C N1(C(C23OCCC(C)(C2)C3)=O)CCC2(C=C(C(=O)NC3CCC(O)CC3)C2)C1 c1(C(N2CC(C)(NC(c3n(CC)ncc3)=O)C2)=O)cc(=O)n(C)cn1 n1(CC(c2ccccc2)OC)c(N2CCC(C3CCCO3)CC2)nnc1CCO c1(C(N2CC(C)C(CNC(=O)C(=O)C3CCCC3)CC2)=O)cc([N+](=O)[O-])cn1C CC(C)CC(O)C(=O)NCC1C2CN(C(=O)CCCOCc3ccccc3)CC12 N1(C(c2c(C)csn2)=O)CCC(C(=O)Nc2cncc(CN(C)C)c2)C(C)(C)C1 N1(C(c2cccc(C)c2)=O)CC(NC(C2CSC2)=O)C2CCCCC12 c1(C(=O)NC(c2cnn(C)c2)CNC(C(CCOC)C)=O)c(C)nc(O)nc1C c1(C(=O)OC(C(C(=O)OCC)=O)C)cnc2c([N+](=O)[O-])cnn2c1 c1(C(C(=O)NC2CCC(NC(c3c(C)ocn3)=O)C2)O)ccc(F)cc1 C1(OC)CN(C(C2(c3ccccc3)CC2)=O)CC1NC(C1(C2CC2)CCCO1)=O C=CC(C)C(C)C(=O)NCC1(O)CCN(C(c2ccc(C(=O)OC)o2)=O)CC1 C1(O)(C(N(CCCNC(N2CCC2)=O)C)=O)CCOCC1.C(=O)C=CCCO C(=O)(CCCCC(N)=O)NCc1cn(C2CCN(C(CN(C)CCO)=O)C2)nn1 c1(C(=O)NCC(C)NC(CC(CC)O)=O)cc2ccsc2[nH]1 c1(CC)noc(C(=O)NCC(C(F)(F)F)N2CCN(C(=O)C=NOC)CC2)c1C C1(NC(c2c(C)nn(CC)c2Cl)=O)CCCCN(C(=O)CC2CCOC2)CC1 c1(N2CCC(C(=O)NC(C3CCOCC3)C=C)C2=O)cc(Cl)ccc1Cl C(=O)(C(=O)CCC(C)C)NCC(CCC)C(=O)NC(C)C1CC1 C(=O)(C1=COCCC1)N(C1CCCC1)CCNC(C1(C)CNC(=O)C1)=O C(C(=O)N=S(C)(=O)c1ccc(C(F)(F)F)cc1)N(c1c(C)cc(C)nc1O)C1CC1 C1(NC(C2(C)ON=C(C)C2)=O)CC2(CNC(c3csc(C(N)=O)n3)=O)CC1CO2 C1(C(=O)N(C)CC23COCC(C2)C3)(COC)CC=CCC1.C12CCCCN1C2=O c1(C(=O)NC(C)CNC(C2CC2c2ccncc2F)=O)coc2c1C(=O)NCC2 C1(CNC(=O)CCN2CCC2)CCCC(CNC(=O)NC2CC=CC2)C1 C1(C(=O)NC2C(NC(c3cnn(CCF)c3)=O)COCC2)CC2(C1)CC(O)C2 N1(C(CCS(CC)=O)=O)CCN(C(=O)CCc2cc(C)cs2)C(C#N)C1 N1(C(C(N)=O)=O)CC2CC2(CNC(=O)CNC(c2ccc(O)cc2)=O)C1 c1(C(CNC(C)=O)NC(C2CCON2)=O)ccc(F)cc1 C1(NC(=O)CC2(O)CC2)CN(C(C2CCCOC2)=O)C2(CCCC2)C1 C1(CCNC(c2nc(CC)sc2)=O)CN(C(=O)CCc2cscn2)CCO1 c1(C(N(CCn2cc(CC3CCCOC3)nn2)CC)=O)nc(Br)n2c1COCC2 Cc1ccc(C(=O)NC2CCC(NC(C3CCC(C)CO3)=O)C2)c(N)c1C CC(CN1CCOCC1)C(=O)N1CCC(C(C)(C)NC(C2CC(=C3CC3)C2)=O)C1 c1(C(N2CCC(N(C(=O)C(C)=C(C)C)CCC)C2)=O)ccc2n[nH]c(C)c2c1Cl C=C(CNC(C1CC(OC(F)F)C1)=O)CCNC(=O)C(C)Oc1ccccc1 N1(C(CCOCCOCC)=O)CCC(N(C)C(C2CCC(C(C)(C)C)O2)=O)C1 CC1c2cc(F)cc(F)c2CCN1C(C1CCCC1c1cccc(N)c1)=O Cc1[nH]c2ccnn2c(=O)c1CC(=O)NCC1(CNC(=O)C(C)(C)F)CC1 c1(CNC(C2C3CN(C(c4[nH]n(C)c(=O)n4)=O)CC23)=O)cccc(S(C)(=O)=O)c1 C(=O)(CCCCCCCCCO)N1C2CC(CNC(C3(C)CCOC3)=O)(OC2)C1 c1(C(=O)NCC2CC(C)(C)CN2C2CS(=O)(=O)CC(=O)N2)ncc2c(n1)COC2 N1(C(C2CCS(=O)(=O)N2)=O)CCC2(CCCN2c2cnc(F)cn2)CC1 c1(C(=O)NC(CC)CNC(c2[nH]c(O)nc2C)=O)cccn2ncnc12 CC1(C)CC2(CCN(C(c3cncs3)C(=O)Nc3ccc4c(c3)OCCO4)C2)CO1 N1(C(C(COCC)n2cc(CO)nn2)=O)CCNC(=O)CC1C.C1C(O)CC(=O)N1 CCCCCCC(=O)NCC1(NC(=O)C=CCN2CCCC2)CCOC1 Cn1cnn(CCC(=O)NC2CC(NC(c3ccon3)=O)C2)c1=O C(c1ccccc1)=CCC(=O)NC1CCC(CNC(C(C)n2cnnn2)=O)C1 c1(C(N2C3CCN(C(C4N(C)C(=O)OC4)=O)CC3C2)=O)cnc2c(c1)nnn2C c1(C(=O)NCC2CCCN(C(=O)C(O)C3CCCC3)C2)ccc2c(c1O)CCC2 N1(C(c2n[nH]c(C)c2Cl)=O)CCN(C(c2[nH]nc3ncccc23)=O)C2CCC12 c1(C(C)C)nc(C(C)C)c(C(=O)NCC2C3CN(C(=O)OC(C)(C)C)CC23)s1 CC1CCCN(C(=O)C(F)=CC2CC2)C1CNC(=O)CNC(=O)C1CC1 C(CCCCC(=O)N1CCCC1CCCNC(=O)C(O)CSC)OC c1(C(=O)NC2C(NC(C3(NC(N)=O)CC3)=O)COC2)ccc(C2=CCCC2)cc1 N1(C(CCCSC)=O)CCCC(C)(C)C1C(=O)NCc1ccnc(C#N)c1 N1(C(C(C)CC2CCCCC2)=O)CCC(C(C)NC(c2cnn(C)n2)=O)CC1 c1(CC(=O)NCC2C(NC(c3nncc(OC)c3)=O)CC2)ccn2cncc2c1 N1(C(CNC(=O)OC(C)(C)C)=O)CCOCC1(C)c1cn(C2C=CCCC2)nn1 C(CC(C)C(=O)NCC1CCCCN1C(c1n[nH]cc1CC)=O)=CCC S(=O)(=O)(c1ccc(F)c(C(=O)O)c1)N1C(C(=O)Nc2cccc(C)n2)CC1 C1(NC(=O)C=CCO)CCCC(NC(c2cc(-c3ccco3)on2)=O)CC1 N1(C(c2c(CCOC)occ2)=O)CC2CC(C)N(C(=O)CCC3CCCO3)C2C1 CC(C)(F)CC(=O)NCC12CC1CN(C(=O)C1CC1)C2 c1(CNC(=O)Cc2ccnn2C2CC2)ccccc1I c1(CC(=O)OCC(=C)CC)c(C)nsc1NC(=O)C1CC1 CC(C)(C(O)C(=O)NC1CC(Cl)(Cl)C1)c1ccccc1 N1(C(c2c(C(C)(F)F)n[nH]c2)=O)CCN(C(C2CCC(C#N)C2)=O)CC1 Cc1cc(Cl)c(C(=O)NC2COCC2NC(=O)CCC(C)C#N)cc1Br N1(C(C2C(C(=C)C)OCC2)=O)CC(NC(=O)C2=CCC2)CC(F)(F)C1 C1(C2CC2)(C(=O)NC(C)CCN(C(=O)CN2CC(=O)N(C)C2=O)C)CCOCC1 C1(NC(C(C)SCC)=O)CCOCC1.C1(C(=O)NCCOC)CCN(C)C1 N1(C(C=C(C)Cl)=O)CC2CN(C(c3sc4ncccc4c3N)=O)CCC2(CO)C1 c1(CNC(c2c(C3CCCN(C(C)=O)C3)n[nH]c2)=O)c(Cl)c(C)nn1C C(=O)(C(C)S(=O)(=O)C(C)C)NCC(CNC(c1c(C)cccc1O)=O)C(F)(F)F CC(CCC(F)(F)F)NC(C1(NC(=O)C=CC2CCCCC2)CSC1)=O c1(C(=O)NCC2(F)CC(NC(C=CCCC(C)C)=O)C2)cnc2cccnn12 N1(C(c2c(CC)ocn2)=O)CCC(c2cn(C3CCCN(C)C3)nn2)CC1 S(=O)(=O)(c1cc(C(=O)OC)c(O)cc1C)N(c1ccc(C#C)cc1)C1CCC1 C(CCN=c1cc(C(C)=O)nc[nH]1)OC1CCN(C(C(CC)n2cncn2)=O)C1 c1(C(N2CCOCC(CC)C2)C(=O)NC(C)(C)C)ccc2nonc2c1 C1(C(N2CCOC(CC3CC3)C2)=O)CCOCCN1C(c1n[nH]c2c1COC2)=O Cc1noc(C)c1C=CC(=O)NCCC1CSCCN1C(c1sccc1C#N)=O C1(CCC)CN(C(c2cscc2Br)=O)CCN1C(c1cccs1)=O c1(NC(C(COC)NC(c2ccnn2C(C)C)=O)=O)ccc(Cl)cc1C c1(CC)occ(C)c1C(=O)N(CCC(C)NC(C12CC(C)(CO1)C2)=O)C CC1=NS(=O)(=O)N(C)C=C1C(=O)N1CCOCC1CNC(=O)C=Cc1ncco1 CCC(C)(C)C(O)C(=O)NCC1(OC)CCN(C(c2c(Cl)nn(C)c2Cl)=O)C1 N1(C(C(COC)C)=O)CCC=C(C(=O)NCC(C)(CO)OC)C1 Cc1oc(C)c(C(N2CSCC2C(=O)NCC(C)(O)C2CCCC2)=O)c1C N1(C(C2CN(C(CC3(OC)CCCCC3)=O)CC2C)=O)CC(CO)CCC1C C1(OC)CN(C(c2cncnc2)=O)CC1C(=O)N(CC(C)C(C)C)C c1(C(C(=O)NC2C(C)N(C(C3CCC3)=O)CC2)O)ccc(Cl)c(F)c1 c1(CNC(=O)CN2CCC(O)CC2)cnn2c1CN(C(C1CSCCS1)=O)CC2 N1(C2CN(C(C(N3CCOCC3)C)=O)C2)CCN(C(C2CC(F)(F)C2)=O)CC1 CON(C)C(=O)C(C)NC(=O)C=C(C)CNC(=O)C=CC(F)(F)F N1(C(C(C)OCC)=O)CC(NC(C2(CN(C)C)CC2)=O)CC(F)C1 Cc1ccccc1-n1nc(CCN(C)C)nc1C1CC(CF)C1 c1(C2N(C(=O)NC3C(c4ccc(=N)[nH]c4)CCC3)CCC2)cc2ccccc2o1 CCC(C)C(C(=O)NCC(C)=CC(=O)N(C1CC2(CCC2)C1)C)OC c1(OC)c(C(=O)N(C)CC2C3CN(C(=O)Cc4ccnn4C)CC23)ccnc1Cl C1(CC(=O)NC(C2CCN(C(C3CC(=O)C3)=O)C2)C)OCCC1(C)C N1(C(C)=O)CCCC12CCCN(C(C1C(CNC(C3CCC(C)(C)C3)=O)C1)=O)C2 C12(NC(C(C)c3cccs3)=O)CCC(CN(C(=O)C(c3ccccc3)O)C1)C2 C=C(C)CCCC(=O)N(CC(=O)NCc1ccc(C)cn1)C1CC1 c1(OC)cc(C)c(C(=O)NCC2(NC(=O)CC(C)(C)C#N)CC2)c(C)c1 CC(CC(=O)N1CCC(n2cc(CNC(=O)C(C)N(C)C)nn2)CC1)C(C)(C)C C1(C(N2CC(CN(C)C(C34CC3COC4(C)C)=O)C2)=O)CC2CC(O)CC(C1)C2 CCCCCC(F)C(=O)NC(CCC)C(=O)NC1CCOC1C c1(OC)ccc(CNC(c2nc(-c3ccncc3)cs2)=O)o1 N1(C(CCC(C)OCC)=O)CCCC(O)(CNC(c2conc2C(C)C)=O)C1 C(CCCC=C)(C(=O)N1CCOC(C)C1)NC(CCSCC#C)=O C(c1cc(F)cc(F)c1)=CC(=O)NC1CC2(C(NC(C(C(=O)OCC)F)=O)C2)C1 O=C(C1=CC2CCC(C1)C2)N1CCC2(CCN(C(c3ccc(O)c(Cl)c3)=O)C2)C1 c1(C(N2CC(N(C(C(CC)c3ccccc3)=O)C)C2)C)ccccc1Br c1(N2CCCC(CCC)C2)nc2c(c(=NC(C)CNC(C)=O)[nH]1)SCC2 Cc1oc(C#N)cc1C(N1CCN(C(=O)CC23CC(C2)C3)C(CC(F)F)C1)=O N1(C(C=CCN(C)CC)=O)CCN(C(=O)C=CC2CCCCCC2)CC(O)C1 C12(C(N(CCOC)CC3CCCC3)=O)CCCC1N(C(C1CC(F)(F)C1)=O)CC2 CN1CCCC(CC(=O)NC2COCC2CNC(=O)C=CI)C1 C(C)(C)(CC(=O)NCC1CCOC1C)N(C(Cn1c(C)ncc1)=O)C N1(C(C(C)OCC(C)C)=O)CC(CNC(=O)CCc2cccnc2)OC(C)(C)C1 C(Cc1ccsc1)CN=c1[nH]c(N2CCC3CCCC3C2)nc2c1CCC2 C(CC(CO)NC(=O)NC(=O)C(c1ccccc1)n1cccn1)OCC N1(C(C2C(=O)NCCCC2)=O)CC2CC1CN(C(C1(C3CC3)CCC1)=O)C2 c1(OC)ccc(OCC(=O)NC2CCCCC2NC(c2cnc(Cl)s2)=O)cc1 C1(C(C)C)CN(C(=O)CC2CC=CCC2)CCN1C(C1CCCC(F)C1)=O C1(C)(NC(c2ccc(C)n2C)=O)CCCN(C(C2(C#N)CCCO2)=O)C1 C1(C(N(C2CCCN(C(C3C(C)CC3)=O)C2)CC2CC2)=O)CC12CCCCC2 c1(C(N2CCC(C3CC3)(NC(CSC)=O)C2)=O)cncc2cccnc12 C(=O)(C1=CC(O)CCC1)N(C)CC1CCC(NC(C(C)N(C(C)=O)C)=O)CC1 C1(NC(c2ccc(C)nc2C)=O)CC2CCC1CN2C(c1cc(N)nc(Cl)c1)=O c1(C(N2C(C)CN(c3ccccc3F)CC2)=O)nc[nH]c2ncc(Br)c1-2 N1(C(C=CC(=O)OCC)=O)CCC2(CCOCC2)C(CNC(=O)C(F)OC)C1 c1(C(CO)NC(C2(CC=C)CCOC2)=O)ccc(Cl)cc1Br C1(C(=O)NC(CCNC(c2c(Cl)cnc(CC)n2)=O)C)Cc2cccnc2C1 C1(NC(c2c(C)n(C(C)C)cc2)=O)CN(C(C2(C#N)CC(C)C2)=O)CCC1(C)C C(=O)(C1=NNC(=O)CC1)N1CC(CCCC)N(C(=O)COC2CCOC2)CC1 c1(-c2c(C(N(CCN(C)C)C)=O)csc2)cc(F)c(O)cc1F C(=O)(CCCC(=O)N1CCCC(CO)(CNC(=O)CCCC2CC2)C1)NC(C)C C1(CC(N2CC(F)(F)C2)=O)C2CCCC2N1C(=O)C=Cc1cnccn1 C#CCC(C)(C(=O)N1CCC1)NC(=O)C=CC=CCC.C1(=O)CN1 N1(C(c2ccc(C)nc2N)=O)CCC2CC2(NC(=O)C2=C(Cl)CC2)CC1 c1(C(N2C(CNC(c3ccsc3C#N)=O)CCC(C)C2)=O)cnc2occc2c1 C(=O)(CC(C)C(C)C(C)C)NC(CC)(CNC(c1c(F)cc(F)cc1F)=O)CC c1(CCC(=O)NC2C(CNC(C(CCCOC)C)=O)C2)ccc2ccccc2c1 C1(n2cc(NC(CCCOC)=O)nn2)CCN(C(=O)CCOCP(C)(C)=O)CC1 C1(C(N2CC(O)(C(CNC(C3(CCCC)CC3)=O)(C)C)C2)=O)C2CCOCC12 Cc1cc(C(=O)NCCC2CN(C(=O)C(F)(F)C(F)F)CC2C)c(C)cn1 c1(CC)nonc1C(=O)N(C1CCN(C(c2cnn(CC(C)C)c2)=O)C1)CC N1(C(C(CCOC)OC)=O)CCN(C(=O)CCC2(C)CC2)CC1COC Cc1cc(CC(=O)NC2CCC(N(C(=O)C=Cc3cc[nH]n3)C)CC2)cc(O)c1 c1(C(N(C2C3CN(C(=O)Cn4ccc(C(F)F)n4)CC23)C)=O)cccc(S(C)=O)c1 c1(NC(=O)NC(C2N(C(C(CC)C)=O)CSC2)=O)cccc(NC2CCC2)c1 Cc1ccc(CC(C)NC2CCC2)c(Cl)c1.c12ccc(cc1)NC(=O)C2N(C)C C(=O)(C(CC)C(F)(F)F)NC(CC)CNC(=O)Cc1cc(C)ccc1C c1(NC(CCCC)CC)cc(=NC2CCc3c(n[nH]c3Br)C2)[nH]c(C(F)(F)F)n1 c1(C(C(=O)N2CC(CCNC(COC)=O)C2)CC)ccc(F)cc1 c1(-n2cc(-c3n(C)cnc3)nn2)ccc(S(N)(=O)=O)cc1 C1(C(N(C(CC(CC)C)C)C)=O)C2CCC(C2)C1NC(C1(COC)COC1)=O c1(CN(C)CCNC(=O)CONC(C2OCCC2C(F)(F)F)=O)cn(C)cn1 Cc1ccc(C(C)CC(=O)NCCOCCN(C(=O)CC(C)C)C)cc1 S(=O)(=O)(c1ccc(Cl)s1)N1CCN(Cc2ccc(C(=O)OC)cc2)C2C1C2 C(N=c1[nH]c(=NCC2CC23CCOC3)[nH]c2c1COC2)c1ccc2c(c1)COC2 c1(C(N2CCCC(CCNC(CN3C(C)CC3)=O)C2)=O)cc(Cl)ccc1Cl CC1CN(C(c2cc(Cl)c(Br)s2)=O)CCN1C(C12CCC1C2)=O c1(N2CCC(NC(=O)CC3CCCCO3)C(F)C2)nc2cc(Br)cnc2s1 N1(C(C2CN(CCC)C(=O)C2)=O)CCCN(C(=O)CNS(=O)(=O)CC)CC1C N1(C(C(c2c(C)n[nH]c2C)C)=O)CCCN(C(=O)Cc2nncn2C)CC1 C(=O)(C1=NOCC1)N(CCN(C(C)C)C(c1cccc(C2CC2)c1)=O)C c1(C(=O)NC(C2(O)CCN(C(c3cccc(C)n3)=O)C2)C)nsc2ccccc12 c1(OCC)ccc(C(=O)N(C(C)CNC(C2CC=CCO2)=O)CC)cc1OC C1(C(N(CCCN(C(=O)C(C)OC2COC2)C)C)=O)CCn2ccnc2C1 C1(C(=O)NCC2(NC(c3cc(OCC)ns3)=O)CC(OC)C2)CCN(C)S1(=O)=O N1(C(c2ccc(N(C)CCO)nc2)CC(=O)NCC)CC(C)OCC1COC C1(C(N(CCC(=O)NC)CC)=O)CC12CC(NC(C1CCCN1C)=O)C2 N1(C(COCC=C)=O)C2CCC(C(=O)NCc3ccc(F)cc3)C1CC2 O=C(C1CCCc2n[nH]cc21)NCC1CCN1C(=O)CC12CCC(CC1)C2 c1(C(=O)NC2CCN(C(C3CCS(=O)(=O)N3)=O)C2)ccc(O)c(Br)c1 C1(NC(CCCc2scc(C)n2)=O)CCN(C(=O)C(=O)NCC2CC2)CC1O CCCCC(CCC)NC(=O)C(C1CCC1)NC(c1coc(C)c1)=O C=CCC(C(=O)N=S(C)(=O)N1CNC2(CCCCC2)C1)c1ccccc1OC N1(C(C2CCCN(CCC)C2)=O)CC(N(C(=O)Cc2cnc[nH]2)C)C2(CC2)C1 c1(NC)cnncc1C(=O)NCc1ccc(C(=O)NCC2CCC(=O)N2)s1 C(CC(O)CC(=O)N1CCC(OCCNC(=O)CC2(C)CCCO2)CC1)SC C1(CNC(C2(CCNC(c3cccc(=O)o3)=O)CC2)=O)CCCNC1=O Cc1ccc(C(N2CCC(C)(CNC(C3CCC(C(N)=O)C3)=O)C2)=O)nc1C c1(C(=O)NCC(=C)CCNC(C2CC2[N+](=O)[O-])=O)noc2c1CC(F)(F)CC2 C1(NC(c2nc(C(C)NC(=O)CN3CC(C)(C)C3)oc2)=O)CCCC1(C)O C1(CC)(NC(=O)C=Cc2cccc(CO)c2)CCN(C(=O)CCNC(C)C)CC1 c1(C(=O)OC)cc(C(=O)NCC#CCNC(=O)C(C)Cc2ccccc2)ns1 C1(NC(c2nc(C)oc2)=O)CN(C(c2cncnc2C(C)C)=O)CCC1C c1(C(=O)NCC(CC)(C)NC(C2CC(F)C(=O)N2)=O)oc(C(C)C)nc1C Cc1ccc(O)c(NC(C2CCC2NC(C2C3CCC(F)(F)C23)=O)=O)c1 C1(NC(C(CC)CC)=O)COCCN(Cc2ccccc2F)C1 C1(NC(=O)CC2CCOCC2)CC2CCC(C1)N2Cc1ccccc1Br c1(N(C)CC)cccc(CNC(CO)C2COC2)c1 C(CCC(C)NC(C1(CCNC(=O)COCCN(C)C)CCC1)=O)=C(C)C c1(NC(CC(=O)NC(C)C)C)ncccc1S(=O)(=O)N1CCOC(C(C)C)C1 C1(C(C)(C)C)CCCC(C(=O)NC2CC(F)(CNC(=O)Cc3cn[nH]c3)C2)C1 C(C)(C(CC(=O)NCCCSC(C)(C)C)NC(=O)C(C)(C)CCOC)OC N1(C(c2c(CC)c(OC)ccc2)=O)CCC2(C1)CN(C(=O)CC(C)C)C2 CC1COc2c(C(=O)NCCC3CN(C(C45CC(C)C4C5)=O)C3)cnn2C1 C1(NC(C(C)OCOC)=O)CC(F)CN(C(C2CC3CC3C2)=O)C1 N1(C(=O)NCc2nc(C)oc2)CCC2(CC1)OC(=O)Nc1ccccc12 C=CCC(F)(F)C(=O)N(C(C)C(N1CCC(O)C(C)C1)=O)C1CC1 Cc1ccc(C(N2CC(C(F)(F)F)CC2CNC(=O)CC(C)F)=O)c(F)c1F C(=O)(C1CC=Cc2ccccc21)NCC(CNC(c1cnc2scc(C)n21)=O)O CC1C(=O)N(CC(N2CC(N(C)C(c3ccnnc3)=O)C(C)(C)C2)=O)C(=O)C1C c1(OC)nccc(C(N2CCC(C)(c3ccc(C)cc3)C2)C(=O)NC(C)C)n1 N1(C(CC(C)(C)C)=O)CCCC(C)(NC(=O)CCCC#N)C1 CCC(CO)N=c1cccc(S(=O)(=O)NCC2(C)CC=CCC2)[nH]1 C(c1ccccc1Cl)=CC.c1(C(C(=O)N(C(=O)CN)CC)=O)cccc(C)c1 c1(C(CO)N(C)C(c2cc(-c3csc(CO)n3)c[nH]2)=O)cccc(Cl)c1 C=CCC(C(=O)N1CC(NC(=O)Cc2cccc(F)c2)C(C)C1)C(C)C CCCC(C(O)C(=O)N1CCCC(O)(CO)C1)NC(=O)C(C)C1(O)CCC1 C1(NC(c2c(C)oc(Cl)n2)=O)CN(C(c2nn(C)nc2C(F)(F)F)=O)CC1(C)C C1(CC)CC(C(=O)NCC(CNC(c2cc(C#N)cs2)=O)OC)CCO1 N1(C(c2c(OC)nccc2)=O)CC2=C(C1)CN(C(c1csc(C3CC3)n1)=O)C2 N1(C(C(C)(C)CF)=O)CCC(NC(c2cc(C3CC3)ccc2F)=O)C(CO)C1 c1(C(=O)NCCN2CCN(C(C3CCC3(F)F)=O)CC2)ccncc1C(F)(F)F c1(C(C)C(=O)NC(C)(C)CCNC(c2csc(Cl)n2)=O)ccc(Cl)cc1 C(N=c1[nH]c(=NCc2nnc3cccnn23)c2ncccc2[nH]1)c1c(N)cncc1 Cc1cc2nc(NC3(CNC(c4ncoc4C4CC4)=O)CCCC3)cc(=O)n2o1 C1(C(COC)=O)CSc2ccccc2O1.c12nnc(C)n1CCS2 N1(C(c2c(C)nsc2)=O)CCCN(C(c2csc3ccccc23)=O)CC1C(C)C N#CC1CN(CC2CCCCN2C(c2ccc(Cl)nc2F)=O)CCO1 c1(C(=O)NCC(CN(C(C2(F)C(C)C2)=O)C)O)sc(Br)cc1F Cc1ccc(O)nc1CNC(Cc1cc(Br)ccc1Br)C(=O)O C(C)(CCN=c1nc2sccc2c(N2CCCC(C)(F)C2)[nH]1)SC C1(NC(c2nn(CC)c(C(F)(F)F)c2)=O)C2CC1N(C(=O)C(C)(C)F)C2C Cc1cc2sc(C(=O)N(CC(C)NC(=O)CCc3cncs3)C)cc2s1 CCC(CCC(C)C)(c1nnnn1-c1ccccc1OC)NCCC(N)=O c1(OC)c(C)cc(C(N2CC3(CNC(C4SCCS4)=O)CCC2CC3)=O)cc1C N#CC1=C(C(=O)N2CC3CC2CN(C(c2ccc(C(N)=O)o2)=O)C3)CCC1 c1(C(N(C)CC2CCN(C(CCCOC)=O)C2)=O)ncccc1Br c12sccc1CC2=O.N1(C(=O)O)CCCC1c1ccc[nH]1 CCCCCC(F)C(=O)NCCC1CC(OC)CN1C(=O)CC(CC)SC N1(C(c2c(COC)cco2)=O)CC(C(=O)NCC2(C(=O)OC)CC2)C(F)C1 C1(OC)CCCCC1NC(=O)COCCNC(C1(O)CCOC1)=O N1(C(c2c(C)ccs2)=O)CCN(C(c2ccc(C(F)(F)F)cc2O)=O)CC1CO N1(C(c2c(C)ocn2)=O)CCC(CNC(c2c(F)cccc2Br)=O)C(O)C1 C1(NC(CCCC(=O)OC)=O)C2CCCN(C(c3cscc3Cl)=O)C2C1(C)C c1(CC)c(C(=O)NCC2CCC2NC(=O)C(C(C)C)C2CCC2)nnn1CC c1(COCCOC)cccc(C(N2CCC(NC(=O)Cc3csnc3C)C2)=O)c1 N1(C(C(COC)OC)=O)C2CCC(C(=O)NCCOCCOC)C1CC2 N#Cc1cc(N2CCOC(c3ccc(Br)cc3)C2)c2ccccc2n1 c1(OCCC)c(NC(=O)CNC(=O)CN(C)C)cccc1C CC(C)C(C(=O)NC(C)C(C)n1cccn1)C(C)NC(c1ccoc1)=O C(=O)(CS(=O)(=O)C1CC1)N1CC(NC(c2c(C)nn(CCC)c2C)=O)C2(C1)CC2 CC1(CNC(=O)Cc2c[nH]nc2O)CCN(C(C2CCCN2C(=O)C2CC2)=O)C1 c1(NC(C2C(C(=O)NC3CCC(OC)CC3)C2)=O)cc(F)ccc1F CS(=O)c1ccccc1C(N1CCN(CCNC(=O)C(F)C(C)(C)O)CC1)=O c1(C(N(C2CCN(C(=O)C=CSC)CC2)CC)=O)ccnc2c1nnn2C N1(C(C2CN(CC(C)C)C(=O)C2)=O)CC2CC1CN2C(c1ccccc1NC)=O N1(C(C2C(C)CCN2C(=O)Cc2cn(C)cn2)=O)CC2CCC(O)C(O)C12 N1(C(Cc2ccc(SCC)cc2)=O)CC(CNC(=O)C(C)O)C2(CCC2)C1 C#Cc1ccc(CC(=O)NC2(C(=O)OC)CC2CC)cc1 C1(NC(C(C)OC)=O)CCCCC1NC(=O)CCNC(=O)CO c1(C(N2CC(C(C)NC(C=CCCC)=O)OCC2)=O)cccc(C(F)(F)F)c1Cl Cc1ncnc(C)c1C(=O)NC(CCN(C)C(C1CC2(CCC2O)C1)=O)C(C)C N1(C(c2cc(NCC)cc(F)c2)C(=O)NCCOC)CC(F)(F)CCC1C C(=O)(CC(C)(O)C(F)(F)F)N1CC(CC)N(C(c2cc3c(nn2)CCC3)=O)CC1 CN(C)S(=O)(=NC(=O)c1cccc(OC(F)(F)F)c1F)N1CCNCC1 C1(C)(CC)CC(C(=O)NC2CC(NC(=O)Cc3ccnn3C)C23CCC3)CCO1 Cc1ccn(CCC(N2CCC(CNC(=O)CC3CCC(=O)N3)C2)=O)n1 Cc1cc(C(=O)NCC(C2CCCC2)NC(C2(Br)CC2(F)F)=O)cnn1 CCC(CC(=O)NCC12CCC(CN(C(c3ns[nH]c3=O)=O)C1)C2)C(C)(C)C S(=O)(=O)(c1cc(Cl)c(Cl)cc1Cl)N1CCC(NC(C2(c3cccc(Br)c3)CC2)=O)C1 C(C(=O)N1CCC(C(N2CCOC(C(N)=O)C2)=O)O1)N(C)C1CC1 C(=O)(CC(C)CCC=C(C)C)NCC1(C(C)NC(CCC(=O)OC)=O)CC1 N1(C(CC(C)C)=O)CC(CNC(c2ccccc2Br)=O)CC1C C(c1cnn(C)c1)=CC(=O)NC(C1CCN(C(C2CCCC(CF)C2)=O)CC1)C N1(C(C(C)c2ccsc2)=O)CC(CNC(=O)C=Cc2cn(C)cn2)CC(C)C1 c1(C(=O)NCC(C)NC(=O)CCN2CCSC(C)(C)C2)cc(O)ccc1Br C1(C(N2CCC(CCCCCNC(C3C(C)C3)=O)CC2)=O)CC1C1CCOCC1 c1(OC)ccccc1C(N1CCOCC1C(=O)NC(c1ccccn1)(C)C)=O C1(C(=O)NC2(C(C)O)CC2)OCCC1CNC(=O)CN1CCCC1 C1(NC(=NCC)NCC(c2cccs2)N(C)C)CC(C)OC(C)C1 N1(C(C(=O)NCCCSC)c2cnsc2)CCC(CCN2CCCCC2)CC1 C1(CCC(=O)N(CCCNC(C2CC2C(F)(F)F)=O)C(C)C)CCC(O)CC1 C(=O)(C(F)C(C)(C)O)N1CC(NC(CC(C=C)C)=O)C(c2ccc(OC)cc2)C1 C1(C(N2CCN(C(CCC)=O)CC2)=O)CC2CCCCC2N1C(=O)CS(C)(=O)=O C1(CC)CN(C(c2cc(CO)ncn2)=O)CC1C(=O)NCCCCN1CCC1 c1(C(N2CC(N(C(Cc3cnc(C)s3)=O)C)C2)=O)c[nH]c2ncc(F)cc12 C1(C(N2CC(NC(c3c(CC)[nH]nc3Cl)=O)C2)=O)CCC(F)(F)C1O N1(C(CSCC#C)=O)CCC(CO)(CNC(C2CC2C(C)(F)F)=O)CC1 C(CCCCC(=O)NCC(C)CC(=O)N1CCC1C(C)O)=CC CCCCCCCC(C)CNC(c1csc(S)n1)=O C1(C(N2CC(NC(c3cc(C)oc3)=O)(CO)C2)=O)CC(O)CN1C CCC(C)(COC)C(=O)N(C1CCCC1)CCNC(=O)C1=CCCC1C c1(C(C)C(=O)NC(CNC(C2CC2F)=O)C2CC2)ccnn1C c1(C(=O)NC2(CNC(C(C3CCCCC3)OCC)=O)CC2)cc(OC)cc(Cl)c1 c1(N(CC=C)C)nccc(=NCC2CCn3cnnc3C2)[nH]1 c1(OC)cc(C(=O)N(C(C)CNC(C2CN(C)C2)=O)C)cc(Br)c1OC CC1CCN(CCC(=O)N(C(C)CN(C(=O)C(O)Cc2ccccn2)C)C)CC1 C1(CNC(CC(C)N(C(CC(=O)OCC)=O)C)=O)COCCN1C C(CCCCC(=O)NC1CCOC(C(C)C)C1)NC(C1N(CC)CC1)=O Cc1cc(C(=O)NCC(C2CCC2)NC(=O)Cn2ccc([N+](=O)[O-])n2)nnc1O CCC(CN(C)C)C(=O)NCCCNC(=O)CC(c1cccc(Br)c1)C N1(CCC=CCC)CC2CCC(NC(c3nnc(O)nc3O)=O)CC2C1 CCCC(CCC)C(=O)N1C(CC(=O)NCC(c2ccsc2)C)C2CCCC12 N1(c2ccnc(SC)n2)CCC2(CCN(C(c3cccc(Cl)c3O)=O)CC2)CC1 c1(CNC(C(=O)N(S(CC)(=O)=O)C)=O)nc(C)c(C)cc1Br C1(C#N)(C(=O)NC2CC(NC(Cc3cncc(C)c3)=O)C2)CC12CCCC2.C1CCCO1 CN1CC(C(=O)NC)NC1=O.c1cccc(F)c1.C12(CCC1)C(=O)NCC(=O)N2 c1(CC)sc(C(=O)NCCOC2CCN(C(C3C(C)C3C)=O)C2)cc1Br C(N=c1[nH]c(N2CCC3(CC(F)C3)C2)nc2c1CSC2)c1ccc(OC)cc1C C1(C(N2CC(CC(=O)N(C)Cc3c[nH]nc3C)(OC)C2)=O)CCCC(O)C1 CCC(C)CCC(O)CC(=O)NCC(C(C)C)NC(=O)CN1CCC(CO)CC1 C1(NC(=O)Cn2cccn2)CC2(CCN(C(C3CC4(C3)CC4(F)F)=O)CC2)C1 c1(N2CC(CNC(c3c(C)nncc3)=O)OCC2)c(C#N)nnc2ccccc12 C1(C(=O)NCC=CCNC(C2CCCC(F)(F)C2)=O)CCCCC12OCCO2 Cc1cc(C(=O)NC2CCN(C(c3ccc(=N)[nH]c3)=O)C2)cn(C)c1=O n1(CCNC(CC2C(C)C2)=O)cnc(C(=O)N(CCO)CCO)c1 c1(COC)ccnc(C(=O)NCCCC(C)NC(=O)Cc2cc(C)on2)c1 C12CCN(C1(C)C)C(=O)CS(=O)(=O)NC2.Cc1nnc(C(=O)NCC)s1.C(C)(C)C C#CC1CN(C(=O)C(C2CCOCC2)C)CCN1C(c1cncc(C)c1)=O C1(C(=O)OC)CCN(C2CCN(C(c3sccc3CN(C)C)=O)C2)CC1 CC1(C)C(n2cc(CC(N)=O)nn2)c2ccccc2N1N(S(C)(=O)=O)C1CCC1 C1(CNC(c2c(C)nn(CCO)c2)=O)CCN(C(=O)Cc2csc(S)n2)CC1C N1(C(CCOC)=O)CCOCC1CN(C)C(C12CC(OC)C1C2)=O C1(CNC(COC2(C)CN(C(C(CC)(C)OC)=O)C2)=O)CC(C)(C)CCO1 c1(C(C)=O)cccc(C(=O)NCCC(C)(C)NC(c2cc(C(N)=O)[nH]n2)=O)c1 C(C(=O)NCc1cn(CCOCCOC)nn1)(C(C)(C)C)NC.C(CCO)S c1(COC)cc(C(N2CCC2Cn2cc(Cn3ccnc3)nn2)=O)ccc1F C(C(=O)NOC1CC1)(C1(C)CC1)NC(CC1CC(=C)C1)=O C1(NC(CC2ON=C(C)C2)=O)(CNC(=O)C(n2ccc(C)n2)C)CC(F)(F)C1 N1(C(C2CN(C(C)=O)C2)=O)CC2CCC(C1)N2C(=O)CSCC1CCCO1 Cc1cc2sc(C(=O)NC(C)CCCNC(c3cccc(Cl)c3F)=O)cc2s1 C1(NC(CC2ON=C(C)C2)=O)C2CC3C(C2)C13C(=O)Nc1cnn(C)c1Cl n1(C(C)(C)C)ncc(C(=O)NC2(C)CC(NC(C3CC4CC4C3)=O)C2)c1Cl Cc1onc(C(=O)NC2CC(F)(CNC(C3CCC3C)=O)C2)c1[N+](=O)[O-] C(C)(C)(C(C(=O)OC)NC(c1ccc(N2CCOCC2)cc1)=O)OC C(=O)(C1CCS(=O)(=O)c2ccccc21)NCCCN(C(=O)C(F)F)CC C1(CCC(C)NC(C2(O)CN(C)C2)=O)(NC(C2CNC(=O)N2)=O)CCC(C)(C)C1 C=C1CC2(C1)CC(C(=O)NCC1(C)CCN(C(C3CC(S(C)(=O)=O)C3)=O)C1)C2 c1(OC)cccc(C(=O)NC23CCC(CC2NC(=O)C(C)NC(N)=O)C3)c1O N1(C(C(c2cccnc2)NC(C(C)n2cccc2)=O)=O)CCCC(O)(C(N)=O)C1 C1(CNC(=O)CSC2CC2)CCCN(C(=O)CCc2nnc(C3CC3)o2)C1 c1(C(=O)NCC(CNC(=O)C(O)C(F)(F)F)C(F)(F)F)c(F)ccc(F)c1Cl Cc1cnnc(N2CCC(CC(N3CCOC(C(C)C)C3)=O)C2)c1C CC1CC(O)CN1C(C1CC(NC(c2ccc(C(F)F)o2)=O)C1)=O c1(C(=O)NC(CC)CNC(=O)C=Cc2cn(C)cn2)cnc(C2CCC2)cc1C c1(CC)ccccc1OCC(O)CNC(C1CC1c1noc(C(F)(F)F)n1)=O C1(C)(CC)CCCCC1C.C(=O)(C(C)(C)C)N1CCC(c2cccs2)NC(=O)C1 c1(OCCCC(=O)N2CC(NC(C(CC)(C)OC)=O)C2)ccc(Cl)c(F)c1 Cc1nc(-c2cccc(Br)c2)ccc1C(=O)N(C)Cc1nnc(C(C)C)o1 C(=O)(C1=C(Cl)CCOC1)N(C(C)C)CCN(C)C(C1COCCN1C)=O c1(C(N2C3CN(C(CC(C)C(F)F)=O)C(C3)C2)=O)ccnc2ccnn12 N1(C(C2(NC(C=C(C)C(C)C)=O)CCOCC2)=O)CC2CCC2(CO)C1 C#Cc1cn(C)nc1C(=O)NC(C1CCCN1C(c1cccc(N(C)C)c1)=O)C N1(C(C(C)(C)C)=O)CCOC(CCCN(C(=O)CC2CC(F)C2)CCO)C1 N12CCC(CC1)CCC(C1CC1)NC2=O.c1(C2C(C)C2)ncc(Cc2ccco2)o1 c1(C(CC(=O)NCCN(C(C2(CCC)CC2)=O)CC)C)nnc(C)n1C CCC(C)(C)CCCC(=O)NCC1CC(NC(c2ccc3cc[nH]c3c2)=O)C1 C(Cc1ccco1)(C(=O)NOCCCC1CC1)NC(c1ccc(C)o1)=O C1(CN=C(NC(C)C)NC(C)(C)C)CC(C)(C)CC(C)(C)C1 C(=O)(C(=O)C(C)N1CC(CO)(OC)C1)OCC N12CCOCC(C1)NC(=O)C2C.c1(C(=O)N(CCCO)C2CC2)ccc(F)cc1 Cc1cccc2oc(C(=O)NCC3(F)CC(NC(c4ccncc4)=O)C3)cc12 c1(C(=O)NC2(CNC(Cc3ccn(C)n3)=O)CCC2)cnc2cccnn12 C(C(F)(F)F)CC=CC(=O)NCC(C)N(C(CC1(CSC)CC1)=O)C c1(C(N2CCN(C3CN(C(C4(C)C=CCC4)=O)C3)CC2)=O)nc2ncccn2n1 N1(C(C(CSC)C)=O)C(CNC(=O)CCc2ccc(F)cc2)CC2COCC12 C(=O)(C1(C)CCCc2ccccc21)N1CC(O)(CNc2nc(C)nc(C#N)c2)C1 N1(C(CNC=O)=O)CC2CC(C(N3CCC(F)(CO)C3)=O)(C2)C1 C1(C)(CC(=O)NC2CC(n3cc(CCC(=O)N(C)C)nn3)C2)CC(F)(F)C1 Cc1ncc(N)cc1C(=O)NC1(CNC(=O)CCNC(=O)CO)CCOC1 c1(CC(=O)NCC2N(C(CC=C)=O)CCC2C)csc2sc(CC)cc12 CC(C)CC(C)CC(=O)NCC(CC(C)C)NC(=O)CCC1CC1 CC(C)(CCCC(=O)NC(CO)CCC1CC1)NC(=O)C(O)C1CC1 C1(C(N(C2CCC(NC(CCC3C(C)C3)=O)CC2)C)=O)CCC2C(C1)C2(F)F CCCC(C(=O)OC)C(=O)N1CC2CC(NC(=O)CCC(C)(C)C)C2C1 Cc1cncc(C)c1C(=O)NCCC1CCN(C(C2(C)CC(C#N)C2)=O)C1 C12(C(N3CC(CCNC(C4COC(=O)N4)=O)(OC)C3)=O)CCCC(=O)N1CCC2 Cc1ccn(CCC(=O)NCCCN(CCCCNC(C2(CO)CCC2)=O)C)n1 N1(C(CCCOCCC)=O)CC(NC(=O)CC(C)O)C2(CCC2)C1 CN(C1CN(C(C2CCCCC2)=O)CCc2ccccc21)C(C1CNC(=O)C1)=O CCC(CC)(CC)C(=O)NC1CCC1NC(c1ccc(O)c(C)c1)=O Cc1cc(C(=O)NC2CCC(NS(=O)(=O)CCCCCl)C2)cc2c[nH]nc12 N1(C(C(N2CCOCC2=O)C)=O)CCC(CNC(C2CCC2C)=O)C12CC2 CC1(C)CC(NC(=O)COC2COC2)CN(C(c2cc(Br)n[nH]2)=O)C1 Cc1c(Cl)cnn1CC(=O)NCC1(C(F)F)CCN(C(=O)CC2(C)CCCO2)C1 C1(F)(CNC(C(C)OCCc2ccccc2)=O)CCN(C(C2CC(F)C2)=O)CC1 CCC(C)C(O)C(C)C(=O)N1CC(C)(C)C1C1CCN(C(=O)C(C)=C(C)C)CC1 n1(CCF)nc(-c2ccccc2)nc1-c1ccc(CC(F)(F)F)cc1 n1(CCCC(=O)NCCN(C(=O)Cc2nnc(S)n2C)CC)cnc(C#N)n1 c1(C(=O)NC2C(C)CCN(C(C(=O)NCC)=O)C2)cccc2nncn12 C(C(F)(F)C(=O)NC1C2CC1N(C(C1CCCOC1C)=O)C2)OC N1(C(C(CC)C)=O)CC2C(NC(c3cnccc3Br)=O)C2C1 c1(OCCC(=O)NCC2C3CN(C(C4(C(F)F)CC4)=O)CC23)cc(F)ccc1F c1(C(=O)OC)ccc(N2CCN(CCNC(C)=O)CC2)nc1C1CC1 N1(C(c2ccc(C)n2C)=O)CCCC2CCN(C(c3cn(C4CC4)nn3)=O)CC12 N1(C(C)C)CC2(CN(C(=O)CCCCNC(N)=O)CCO2)C1 O=C1NCCOc2c1cc(Br)cc2S(=O)(=O)N1CCC(O)C12CCC2 c1(C(=O)NCC2CCCN(C(CCC#CC)=O)C2)c[nH]nc1[N+](=O)[O-] C=CCC(C)(CC)C(=O)N1CC2C(C(=O)NC(COC)CCOC)C2C1 C(=O)(CC(C)CC(C)C)N1C(CNC(CC(CC)SC)=O)CC(C)(C)C1 c1(C(=O)NC2(C(N3C(C)CC(O)C3)=O)CCN(C)C2)cc2ccccn2n1 c1(OCC)ccc(C(=O)NCCC2CCN(C(=O)C(C)C)CC2)cc1[N+](=O)[O-] N1(C(C2(C)CC(F)(F)C2)=O)CCC(NC(c2sccc2C#N)=O)C(F)C1 N1(C(c2ccc[nH]2)=O)CCC2(CC1)CC(N1CC3(CCCC3)C1)CO2 Cc1ccc2cc(C(=O)NCCN(C(=O)C(c3cncc(F)c3)C)C)cnc2c1 C1(CNC(C(C(CC)O)C)=O)(NC(=O)C2=C(C)OCC2)CC2CCC1CC2 CN=c1[nH]c(C(=O)NC2CC(CNC(=O)C(C)Sc3cccc(C)c3)C2)cs1 CC1(CNC(c2cnc(C3CC3)[nH]2)=O)CCCN(C(C2(C3CC3)CC2)=O)C1 N1(C(CCCN(C(=O)OC)C)=O)CC2CC(CNC(c3cnco3)=O)CC1C2 c1(C(=O)NC2CCC(NC(c3nc(C)nn3C)=O)C2)ccc2c(c1)COC2 c1(C(C(=O)NCC)N(CCCC)CCCC)cnn2cc(Br)ccc12 CC(C)CC(C)C(=O)N1CCN(C(=O)COCc2nc[nH]n2)C(C2CCC2)C1 C1(CNC(c2c(NC)cnnc2)=O)CCN(C(=O)OC(C)(C)C)C(C)C1 Cn1ccc(C(=O)NCC2CCN(C(=O)CC3CCCC3O)C2(C)C)c(O)c1=O C(=O)(C1=CCC(C)CC1)NCC1N(C(c2cc(CC)c(OC)cc2)=O)CC(F)C1 c1(C(=O)NC(CC)CN(C(=O)CCC2CC2)CC)c(C(F)F)nn(C)c1C C1(CC)CCN(C(C2CN(C)C2)=O)C(C(=O)NCC2COCC2(C)C)C1 c1(C(=O)NC2CCC3CN(C(CCOC)=O)CC3C2)cc(O)c2[nH]c(C)nc2c1 N1(C(C(C=C)O)=O)CC2CCCC2(CNC(c2scnc2C2CCCC2)=O)C1 N1(C(C2(CC#C)CC=CCC2)=O)CCN(C(c2cc(CC)no2)=O)CC1C C1(CC(=O)NC(C2CCCN(c3cc(OC)ncn3)C2)C)OCCCC1(C)C C1(NC(C(C2(OC)CCCCC2)(F)F)=O)CCCN(C(=O)C(CO)N(C)C)CC1 C=C(C)CC(C(=O)NC1COCCN(C(=O)CNC(=O)CC(C)C)C1)NC(C)=O C=CC1(C(=O)NC(C2CCCN2C(=O)C(C)Cc2ccccc2)C)CCC1 C(=O)(CCC(=O)NC(CNC(=O)CSc1ccncc1)CO)N(C(C)C)C C1(CNC(CN(C2CCCC2O)C)=O)CN(C(=O)C=Cc2cocn2)CC1C C1(C(N(C(C)CCNC(C2(C)CCC2)=O)C)=O)CC12CCOC2 CC(C)(CC(=O)NC1(CO)CN(C(=O)CCSc2ccc(F)c(F)c2)C1)C(F)F C12(C(N3C(C)CCC(NC(=O)C4=CCCOC4)C3)=O)CCC(C(F)F)(CC1)CC2 C1(C)(CC)CC(NC(=O)CC(CNC(=O)C(C(C)(C)C)OC2CC2)OC)CCO1 C1(NC(C23C(CN(C(CC)=O)C2)C3)=O)COc2ccccc2NC1=O c1(C(=O)NC2CC(CCC(=O)NCC3N(C)CCC3)C2)cccc(O)n1 CN1CCCCC1CC(=O)NCCC1CN(C(=O)CC(F)(F)Cl)CCO1 C1(C(N(CCN(C(COCCC(C)C)=O)C(C)C)C)=O)CCC=CCCC1 N1(C(c2ccc(C#C)cn2)=O)CCCC12CCCN(C(C1(CO)CC1(F)F)=O)C2 C(=O)(CCCC(F)(F)F)NCCc1c(CNC(C(COC)(C)C)=O)nco1 Cc1cn2cc(C(N3CCC(O)(CNC(=O)C(F)C(C)C)C3)=O)cc(F)c2n1 c1(OCC)ccc(-c2nc(C(c3nnnn3C)Nc3ccsc3SC)co2)cc1 c1(SC)cncc(C(N2CCCCC2C(C)NC(c2cnn(C)n2)=O)=O)c1 Cc1ccc(C(=O)NCC2CN(C(c3cc(C#N)c[nH]3)=O)CCCO2)c(O)c1C N1(C(c2scc(C)c2C)=O)CCN(C(=O)C(C)n2cccc2)C(C)C1 C(=O)(C1=CC(C)(C)C1)NC(C)C(C1CCN(C(C)C)CC1)NC1CCCCC1 CN1C(=O)C(=O)N(CC(=O)NCC(C2CC2)NC(C2CCO2)=O)C1=O O=C(NNc1c(Cl)cc(F)cc1Cl)c1cc2ccc(F)cc2[nH]1 C1(F)(CNC(C2(CO)CC2)=O)CCCN(C(C2(CO)CC2)=O)CC1 c1(C(=O)NC(CNC(CCOCC#C)=O)CC)ncccc1S(C)(=O)=O N=c1nc(CCC(=O)NCC2CCN(C(=O)CSc3ccccc3)C2)[nH][nH]1 C#CCCCCCC(=O)N1CCOC(C(=O)NCC2(C)CCCCO2)CC1 Cc1c(Cl)c(C(=O)NC(C2CCCN2C(=O)CCC(=O)c2ccc[nH]2)C)nn1C C1(NC(c2nc(C(C)C)oc2)=O)CC2CCC1N2C(c1cnn[nH]1)=O C1(CCCNC(c2nc(C(C)OC)oc2)=O)CN(C(c2ccc(C)o2)=O)CCO1 C1(NC(c2cncc(SC)c2)=O)CC2(CCN(C(c3n[nH]cc3Cl)=O)C2)C1 C12(CNC(C3CC3c3ccccc3)=O)CCCC(CN1C(C1CCS1(=O)=O)=O)C2 C(CC(=O)N1CCC(N2CCC(O)C2)C1)(c1ccccc1)NC(=O)OC(C)(C)C C1(NC(C2(C)CCCO2)=O)CC2CCC(C1)N2C(=O)Cc1csc2ccccc12 c1(C(=O)NCC(=O)NC2CC(NCCO)C2)cccc(-n2cccn2)c1 CC1OC2(C(=O)NC3CN(C(=O)C(C)(C)C(F)(F)F)CC34CC4)CCC1CC2 CCC(C)(C(=O)NC1CCN(C(=O)CC2(C)CCC2)CC1)C(F)F N1(C(c2n[nH]c(C)c2O)=O)Cc2n[nH]cc2C1C(=O)NC1CCn2cncc2C1 C1(C)(NC(C(C)NC(C2(COC)CC=CC2)=O)=O)CCCCC1C c1(C(N2CC(NC(CC(CC)C3CCC3)=O)C2)=O)ccc(C(F)F)c(C)c1 c1(C(=O)NCC2(F)CN(C(C(CC)OCC)=O)C2)ccc(F)c2occc12 C12(C(N(C(C)CC3CC3)C)=O)CCC(CN(C(C3(C)CC3(F)F)=O)C1)C2 c1(CCC(=O)NC2CCC(NC(C3COC(=O)N3)=O)C2)ccc(O)nc1 N1(C(C2C(CNC(C(CCN(C)C)O)=O)CC2)=O)CC2(CCC1CO)CC2 C(=O)(C1SCCc2ccccc21)N1CCCC(N(C(CCCCCOC)=O)C)C1 CCC(CO)(C(=O)NC1C=CCC(C(N2CC(CO)C3(CC3)C2)=O)C1)OC c1(C(=O)NC2CC3(C(NC(C4C(CC)C4)=O)C3)C2)cc2nccnc2cc1C c1(C(=O)NCC(N(C(CC2C(C)C2)=O)C)C2CC2)c(O)ccc(Cl)c1O C(=O)(C1=CCCC(C)(C)C1)N1C(CC)C(NC(=O)C(C)(CC)CC)CC1 C1(C(C)(C)C)(CNC(COCC(C)C)=O)CCN(C(C2CC2C(N)=O)=O)C1 N1(C(C(F)=C(C)C)=O)C2CCCC1CN(C(c1ccc(N)c(F)c1)=O)C2 C1(C(=O)NC2(C(C)C)CCC2)CC=CCC1NC(c1cnnn1C)=O c1(C(N(CCN(C(=O)C=CC2CCC2)CC)CC)=O)ccccc1OCC(F)F c1(NCC(F)(F)F)ncc(-c2cccnc2C(=O)NCc2cn(C)nc2)cn1 Cc1csc(C(N2CCC(NC(c3ccoc3)=O)CC2)=O)c1Br c1(C(C)C)cc(C(=O)NCCC2CC(C)(C)CO2)c(C(C)C)[nH]1 c1(NC(C2CN(Cc3c(F)cccc3I)CCS2)=O)ccc2c[nH]nc2c1 c1(OC)ccc2ncnc(NCC34CCC(CNC(C)=O)(CC3)OC4)c2n1 N1(C(c2ccc(OC)o2)=O)CC(NC(=O)CSCc2ccccn2)C2(CC2)C1 C(=O)(C(C)(CSC)NC(C1C2CCCCC12)=O)NC1(CCOC)CC1 C(=O)(C(O)C1=CCCCC1)NC(CC(C)(C)C)C(N1CC2(CCC(O)CC2)C1)=O c1(C(=O)NC(CC)(CNC(=O)C2=NOCC2)CC)cc(C#N)cc2ccccc12 N1(C(c2c(CCC)occ2)=O)CCOCC(CNC(=O)C(C)Cc2cnc[nH]2)C1 C1(CCNC(=O)CC2(NC(C3CN4CCC3C4)=O)CC2)CCCCC1O C(=O)(C(C)S(C)(=O)=O)NC(CSCC)C(=O)NCCN(C)C Cc1ccc(CCNC(C2(NC(c3ocnc3C)=O)CC2)=O)nc1 c12ccc(Br)nc1NC(=O)N1C(CC(=C)C1)C(=O)N2.c1(NC)cc(Cl)ccc1Cl C1(N(C(C2(C(=O)Nc3n(C(CC)C)ncc3)CC2)=O)CC)CCN(CC)CC1 c1(CCC(N2C(CNC(=O)CC3CC=CC3)CC2)=O)cc(F)cc(Br)c1 c1(SC(C(=O)N(CCC(C)NC(=O)CCNC(N)=O)C)(C)C)ccc(F)c(F)c1 C#Cc1ccc(C(N2CCOC(C(=O)NC(C=C)C(F)(F)F)CC2)=O)c(C)c1 CC(CN(C)C)C(=O)N1CCC1CNC(C1CCC(c2ccccc2)O1)=O C(c1ccccc1F)=CCC(=O)NC1C=CCN(C(c2cnn(CCO)c2)=O)C1 C#Cc1cccc(CC(=O)NCC(c2cccc(Cl)c2)NC(C2CC(=C)C2)=O)c1 C12(C(=O)NCC3CC(NC(c4scc(C)c4)=O)C3(C)C)C3C4C1C1C2C3C41C C(=O)(C(C)(C)c1ncco1)NC(C1CCOC1)CNC(CC=C(C)C)=O C1(C(N2CCN(C(=O)CC3CCCOCC3)CC2)=O)C2CC(F)(F)CC12 c1(CC(N2C3CC(NC(CN(C)CC)=O)C(C3)C2)=O)coc2ccc(C)cc12 c1(CC(=O)NC2(CNC(C(COCC)C)=O)CC2)ccc(O)c(OC)c1 c1(N(C(CC2(N)CCC2)=O)C(C2CC2)C2CC2)cccc(N2C(=O)CCC2=O)c1 n1(Cc2c(C)noc2)cnnc1S(=O)(=O)C(C)(C)C C1(C(=O)NC2CC(CNC(C(C)C3CC3)=O)C2)CC2C=CC1O2 C1(C(N2CCC(c3ccc(C)s3)C2)Cc2cnnn2C2CC2)CCS(=O)(=O)N1C CC(CN(C(=O)C(c1cncn1C)O)C)C(=O)NOC1CCCCC1 c1(C(N2CCCC(O)C2C)C(=O)NC)nc(OC)ccc1F c1(NC(CCOCCOCCOCCOCC#C)=O)ccn(C)c(=O)c1 N1(C(C(c2ccccc2)NC(C2CCCCC2F)=O)=O)CCN2CCC1CC2 C(=O)(C(F)(CC)C(=O)C(COC)=O)NCC1(CN(C(CCNOCC)=O)C)CC1 c1(-n2cc(CN(C3CC(=O)NC3=O)C)nn2)cc(C(=O)O)cc(F)c1 C(=O)(C1=NN(C)C(=O)CC1)NC(CC)CCC(=O)NC(C)C(F)(F)F CCC(O)C(C)C(=O)NCCC1CCN(C(C2(c3ccccc3F)CC2)=O)CC1 C(CCCCC(=O)NCCC1CCCCC1)NC(C1C(C)=CCS1)=O CC1CC(C(=O)NCC(C)CC(=O)NCCN=S(C)(C)=O)CC(=O)N1 C12(C(N3CCC(N(C(=O)C(F)C4CCC4)CC#C)CC3)=O)CCCCC1OCC2 C1(CC(N)=O)(NC(Cc2c(C)occ2)=O)CCN(C(C2CCC2C(N)=O)=O)CC1 Cc1cccc(CN(CC(=O)N(C(C2CC3CCC2C3)=O)C2CC2)CCN(C)C)c1 Cc1sc(=O)n(CC(=O)NCC2C(C)CCN2C(=O)CC2OCCC2C)c1C CCCC(C(=O)NC(C)(CNC(c1ccc(C(N)=O)nc1)=O)C(C)C)NC(N)=O C1(CNC(C(C)C(C)(C)C)=O)CC2(CCC2)CN1C(c1cnc2c(c1)COC2)=O Cc1cc(C(=O)Oc2ccc(C)c(OC)c2)nc(CC2CC2)n1 N1(C(C2(CNCc3ccc(OC(F)(F)F)nc3)CC2)=O)CC2CCN(CC)C2C1 c1(N2C(C3CCN(C(C=COCC)=O)C3)CCCC2)cc(C)nc(C)n1 c1(OC)ncnc(OC)c1C(=O)NC1CCN(C(=O)CC2SC(=N)NC2=O)C1 N1(CCC(=O)Nc2ncccc2I)CCC(O)(Cc2ccc(F)cc2)CC1 c1(C(=O)NCCC(C)N(C(c2c(CC)cno2)=O)C)csc(S(N)(=O)=O)c1 N1(Cc2ccn(CC)n2)CCCC(C)(CNC(=O)CCc2ccncc2)C1 c1(C(N2CCC(OCCNC(=O)C(=O)NC3CC3)C2)=O)ncn2c1CCC2 c1(C(=O)NCCN(C(=O)C(C)(C)C(F)F)C)cnn2c1OCC(O)C2 c1(C(=O)Nc2ncc(OC(C)C)nc2)cc(F)ccc1F C(CCCCCNC(=O)Cn1ccc(Br)n1)NC(c1cn(CC=C)nc1)=O C1(C(N2CCCN(C(c3cnn(C(C)C)n3)=O)CC2)=O)CCN2CCCC2C1 C(C(C)CC(=O)N(C)CCc1cc[nH]n1)NC(Cn1ccc(C)n1)=O CC(C)C(C(=O)NCC1CC(F)CN1C(=O)C=Cc1cn(C)cn1)c1cc[nH]n1 C12(NC(c3cncc(OCC(F)F)c3)=O)CC3CCC(C1C2)N3C(=O)CC(F)F c1(OCC(=O)NCC(C)NC(C=CSC)=O)cccc(C(C)(C)C)c1 C1(CS(N)(=O)=O)CN(C(=O)CCc2cnc(O)[nH]2)CCO1 CCCCN=C(NCc1cc(C)ns1)N1CCC(C)(OC)CC1 C1(C(=O)NC2C(C)CN(C(=O)COCCCN=[N+]=[N-])C2)CCn2cnnc2C1 C1(C(NNC(c2c(C)ncn2C)=O)=O)COCCC1C1CC1 c1(C(CC(N2CCC(N(C(C)=O)Cc3cnc(CC)s3)C2)=O)C)c(C)n[nH]c1C Cc1ccc2c(NC3CCc4ncc([N+](=O)[O-])cc4C3)ncnc2c1Br N1(C(N)=O)CC(O)CC1C(=O)NCCCn1cnnc1-c1ccccc1 Cc1cccc2[nH]cc(C(=O)NC3CC3CNC(c3ccc4nn[nH]c4c3)=O)c12 C1(C(=O)NCC(CNC(c2cnn(C(C)C)c2Cl)=O)C)CCC(C)(C)CO1 Cc1ccc2[nH]nc(C(=O)NCCOCCNC(=O)C#CC3(C)CCCO3)c2c1 C1(OC)CC(CNC(=O)CCc2c(C)noc2Cl)N(C(=O)CC(C)OC)C1 C1(C(N2C(CCOC)CCC2)=O)CCCN1NC(=O)c1cc(C2CC2)on1 CC1CN(C(C2(N(C)C)CCC2)=O)CCN1C(c1nnn(-c2ccccc2)n1)=O C=CC1(CNC(C2(CCNC(C3CC(OC)C3)=O)CCC2)=O)CCC1 c1(N(C(N2CC3(C(C(=O)OC)C3)C2)=O)C)c(C)cccc1C c1(CCCC(=O)NCC(C)CNC(C2(O)CCC2)=O)nc2ccccc2[nH]1 CC1CN(C(=O)Cc2ccoc2)CC(C)CN1C(=O)CCc1ccon1 C12(C(=O)NC(C(=O)N(CC#C)CC=C)CCOCC)CCC(C)(C1)OC2 CCC(C)(C)CC(=O)NCC(C1CCCC1)NC(=O)C1=NOC(C)C1 N1(C(C2CC(OC)C2)=O)CCC(C(C)(C)NC(c2ccnn2CC(C)C)=O)C1 Cc1ccc(F)cc1CNC(=O)CCN(C(=O)C=Cc1cscn1)C CCCC(CC)C(=O)NCC1COCCN1C(c1cc(CC2CC2)on1)=O c1(C(N2CC(CNC(c3c(CC)nccn3)=O)OCC2)=O)c(CC)nc(C)n1C c1(C(=O)NCC2C(NC(c3c(C)ccc(Cl)c3)=O)C2)cc(C)c2c(O)n[nH]c2n1 C1(C(=O)NCC(CC)N(C)C)CCC(C)(C)N(C(c2cc(C)n(C)n2)=O)C1 c1(C(c2nnnn2CC)NCCC(CCC)C)cc(C2CC2)ccc1Br CCCCCC(CCC)(c1nnnn1C(C)C)NCCCOc1ccc(Br)cc1 C1(NC(C(C(C)C)NC(C)=O)=O)COCCN(C(=O)CC2(C#N)CCCCC2)C1 Cc1cc(C(=O)NC(C)(C)CNC(=O)C(C)N(C)C)c(N)c(Cl)n1 C1(NC(c2n(CCC)ncc2)=O)(CO)CCN(C(=O)Cc2nncn2C(C)C)C1 C1(CC(=O)NC(C(=O)N(C)CC)C)CCCC(NC(=O)C=C2CCC2)C1 CC1(C)CCC(O)(CNC(=O)CC(C)(C)NC(=O)CC(O)C2CCCC2)C1 c1(C(=O)NCC(C)(C)OCC(=O)Nc2nc(C)nc(Br)c2)c(F)cc(Cl)cc1F Cc1ccc(C(N2C(C(N3CC(N4CCCC4=O)C3)=O)CC(C)(C)C2)=O)cc1C c1(C(=O)NCC2(NC(CC(C=C)C)=O)CCOC2)ccnc2[nH]ncc12 C1(NC(c2nccs2)=O)CN(C(=O)Cc2cnccc2Cl)Cc2nccn2C1 S(=O)(=O)(c1cccc(C(=O)OC(C)=O)c1)N(CCCCCC)C(CO)C(C)C N1(C(c2cccc(O)c2)=O)CCCC(n2cc(CNC(C3CC(O)C3)=O)nn2)C1 N1(C(CCNC(=O)OCC)=O)CCC2(CC1)COC(C)C2NC(=O)C(C)S C1(C2(CNC(COCCCC#C)=O)CC2)CCCN1C(c1cnc(C(C)C)s1)=O C1(CNC(CN2C(C)CC2)=O)(CNC(=O)C(C)Cc2cccnc2)CCCCC1 N1(C(C2OCC(C)(C)C2)=O)CCN(C(C2(Br)CC2)=O)C2(CCC2)C1 n1(CC(=O)N2CC(c3c(F)ccc(F)c3Br)C2)nc2n(c1=O)CCOC2 C(=O)(C(C)(C)CC(C)(C)C)NCC(C1CC1)NC(COc1c(C)c(Cl)ccc1)=O c1(CC(=O)NCCN(C(CCC=CC)=O)CC(C)O)c(OC)cccc1F C1(C(N2CC3CN(C(C(C)C(C)(C)C)=O)CC3C2)=O)CCC2CC(C)CN2C1 C1(C)(CC2(C)CN(C3(C(CN4C(C)CCC4)O)CC3)C2)CC=CCC1 C12(CNC(C(C(C)(C)C)O)=O)CN(C(c3cccc(C(F)F)n3)=O)CC1CCO2 N1(CC(=O)NC2CC(NC(C3CNC(=O)O3)=O)C2)CCc2ccccc21 C(=O)(C(F)(F)Cc1ccc(F)cc1)NCC(C)(C)NC(C(C)n1cccc1)=O N1(C(C(OC)OC)=O)CCC2(CC1)CC2CNC(c1cccnc1)=O N1(C(C2(COC)CC2)=O)Cc2ccccc2C(CNC(=O)CCCN=[N+]=[N-])C1 C1(NC(c2nc(C(C)OC)sc2)=O)CCCN(C(=O)C2CC2)CCC1 N1(C(c2c(OC)csc2)=O)CCC2(CC1)CC2CNC(=O)Cc1cccnc1C N1(C(C2=C(C)CCC2)=O)CCCC12CCCN(C(=O)C1=CS(=O)CCC1)C2 CS(=O)(=O)C1CCCN(C(C2CC(F)CN(Cc3ccc(CO)o3)C2)=O)C1 Cc1nn(C)c2c(NC(C)CCCO)nc(N(C)CC3CC3(F)F)nc12 c1(OCC)ccc(NC(=O)CCc2cc(N(C)C)n(C)n2)cc1 C1(C(=O)NC2C(NC(c3c(CC)non3)=O)COC2)Cc2cc(F)cc(F)c2O1 C1(CCCCNC(C2N(CC)CC2)=O)CCN(C(C2COCCN2CC)=O)CC1 CN1CCCC(NC(=O)C(C2(O)CN(C(=O)CCC3CCC(=O)C3)C2)F)C1=O n1(CC)nnc2c1CCC(C(=O)NC1CC(F)CN(C(C34CC(C)(C3)C4)=O)C1)C2 C1(CC)CN(C(c2cn(C3CCC3)nn2)=O)CCN1C(=O)C(c1cccnc1)C C1(c2n(-c3c(C)cc(C)cc3C)nc(-c3nccs3)n2)CCc2nnn(C)c2C1 c1(C(=O)NCCCN(C(=O)CN2CSCCSC2)C)ccccc1C(C)(F)F c1(C(N2CCC(O)(c3ccc(Br)cc3)CC2)=O)cc(Br)ccc1O c1(CN(CCOC)CC)ccc(OC)cc1.C1CCN1C.C1(=O)CN1 C1(CNC(=O)C=CC(=O)NC2CC2)CN(C(C2CNC(=O)C2)=O)CC1(F)F C1(CC)(NC(=O)Cc2ccc(C)c(O)c2)CCCN(C(=O)C(F)C2CCC2)C1 Cn1c(=O)n(C)c2cc(CN3C4CCC3CC(NS(=O)(=O)C(Cl)(Cl)Cl)C4)ccc12 c1(CC(=O)N(C(CNC(c2c(OC)noc2C2CC2)=O)C)C)ccc(O)c(Cl)c1 C1(NC(CN(C2CCCC2)C)=O)CC(C(F)C(=O)NCCN=[N+]=[N-])C1 C1(CNC(c2n(CC)cnn2)=O)CCC(C)CN1C(c1csc(C2CC2)n1)=O c1(C(=O)NCC(C)N(C)C(c2ncn3c2CCC3)=O)c(N)cc(Cl)cc1F c1(N(C)CC2CC2)ccc(S(=O)(=O)NCCCc2ccc(F)cc2F)cn1 C(=O)(CCCC(=O)N(C)C)N(C1C(NC(c2c(CC)nc[nH]2)=O)CCCC1)C c1(C(N(C(CNC(C(CC=C)C)=O)C)C)=O)nnn2cc(C)nc(O)c12 c1(OC)ccc(C)c(C(N2CC(C)CCC2CNC(c2ccc(Cl)o2)=O)=O)n1 N1(C(C2(S(C)(=O)=O)CCC2)=O)CCC(C2(NC(C3CNC(=O)C3)=O)CC2)C1 N1(CC(=O)N(CCC(=O)NC2CC2C)CC#C)CCC(OC)C1 c1(C2CN(CC(CN(CCC#N)C(C(C)(C)C(=O)O)=O)OC)C2)ccccc1C c1(CC(=O)NC2(C)CN(C(=O)OCCC)C2)ccc(F)cc1 N1(C(c2ccc(C#C)cc2)=O)CCC2CN(C(c3ccc(F)nc3C)=O)CCC12 c1(C(N2CCC(C)(NC(CCNC(=O)NC)=O)C2)=O)cn2cc(C)sc2n1 c1(C(=O)NC2C(CNC(C3C(C=C)CC3)=O)COC2)ccccc1C(C)=O Cc1cnc(NCCCc2nccs2)c(S(=O)(=O)N2CCCC(F)(CO)C2)c1 O=C(N=S(=O)(c1ccc(F)cc1)C1CC1)c1ccc(C(c2ccccc2)O)cc1 CCCCC(CC)CCC(CNC(=O)N(C1(C)CCS(=O)(=O)C1)C)CC C(=O)(C(F)(F)CCn1ccnn1)N1CC(NC(C2CC2[N+](=O)[O-])=O)C1 N1(C(C2(CF)CC(=O)C2)=O)Cc2occ(C(=O)NCC3CCCNC3=O)c2C1 C1(NC(C2(OC)CCOC2)=O)CC2(C(=O)NCC(C)CC(C)C)COC1C2 CC1OCCC1C(=O)NCC(C1CCCC1)NC(=O)C(F)(F)c1ccsc1Cl c1(CC)nn(C)c(CC(N2CC(NC(C3CCC(=O)N3)=O)C(C)C2)=O)c1Br C1(O)(C(N2CC(N3C(=O)CCC3=O)C2)=O)CCN(CCC(F)(F)F)CC1 c1(C(=O)NC2C(CNC(c3c(C)cc(C#N)cc3)=O)C2)ccc2c(c1)COCC2 c1(CNC(C(=O)NCC(C)(CN(C)C)OC)=O)ccc(C(F)(F)Cl)cc1 N1(C(CNS(CC)(=O)=O)=O)CC2CCC1CN2C(C1CCCCS1)=O C1(C(=O)NC2(COC)CN(C(C3CCC(C(C)(C)C)O3)=O)C2)CC2CCC1CC2 C(=O)(C(C)C(=O)N1CCOCC1CC(N1CC(COC)C1(C)C)=O)OC S(=O)(=O)(c1ccccc1[N+](=O)[O-])NC(C)C(=O)NC1CC(F)(F)CN1 C1(NC(c2cnc(C(C)C)[nH]2)=O)CCCCC1NC(c1ccncc1Br)=O O=C(COc1cccc(Cc2ccc(Cl)cc2)c1)NNC(=O)C1CCOCC1 C1(CNC(C(C)n2cncn2)=O)CN(C(C2(C(F)F)CC2)=O)CCN1C c1(C(N2CC(C(N3CCOC4CC34)=O)C2)=O)cccc(I)c1F C1(c2nccs2)(CCNC(=O)NCCC(C)NC(=O)O)CCCCC1.C(C)(C)C Cc1coc(C)c1C=CC(=O)NC1(CNC(C23C=CC(CC2)C3)=O)CCOC1 CCCC(O)(CCC)CC(=O)NCCN(CC(C)O)C(=O)CC1CNC(=O)O1 C1(OC)CC(CNC(c2nc(N(C)C)nc(=N)[nH]2)=O)N(C(C2CC=CCC2)=O)C1 Cc1ccc(=NC(=O)C(=O)NCCc2ccoc2)[nH]n1 N1(C(C2CC(=C)C2)=O)CC2CC(CNC(c3cnc(COC)s3)=O)CC1C2 c1(OC)cccc(OC)c1C(=O)NCC1(NC(=O)C(C)P(C)(C)=O)CCOCC1 C(C(C)(CC)C(=O)NC1CCCC1(C)N(C)C)NC(C(C)OCCOCC)=O C1(c2ccc(C(C)C)o2)CCOCCN1C(=O)C(CN)CN1CCCS1(=O)=O C1(OCC(F)F)CC2CCC(C1)N2c1cncc(C(F)(F)F)n1 N1(CC)CC2C3CCC(C3)C2(C)C1.c12ccc(cc1)c1nnc(n1CC(C)C)s2 c1(C(=O)OC)ccc(NC(=O)N(C)Cc2nc(=O)o[nH]2)cc1OC c1(C(N2CC3C(CNC(c4cc(Cl)c(Cl)s4)=O)C3C2)=O)nnn2ccccc12 c1(CC(=O)NC2(C)CN(C(CC(C(CC)C)O)=O)C2)ccc2c(c1)OC(F)(F)O2 c1(C(N(CCNC(CC(=O)NCC)=O)CC)=O)cc(C)c2n[nH]cc2c1 c1(C(C)SC(C(C)C)C)nc(C2SCCc3ccccc32)no1 C1(O)(C(=O)OC)CCN(C(c2sc(Cl)cc2Br)C(=O)Nc2ccccc2C)C1.C1CC1 O(N=C1CCCCCC1)CC(=O)NC1COCCN(C(c2cnn(C)c2Cl)=O)C1 C1(NC(C2(C)CC(NC(c3ncn(C)n3)=O)C2)=O)CCC(F)(F)C1 N1(C(CCCc2scc(C)n2)=O)CCCN(C(=O)Cn2nc(C)nc2C)CC1C C1(NC(C=Cc2ncc(C)[nH]2)=O)(CO)CCCN(C(C2CCS(=O)(=O)C2)=O)C1 C1(C(=O)NCC(C2CC2)NC(=O)C(C#N)C2CC2)(OC)CS(=O)(=O)C1 c1(C(N2CCN(C(C=CC(=O)NC3(CO)CCCO3)=O)CC2)=O)cc(F)cc(Cl)c1 N1(C(C(C)SC)=O)CCC2(CCCN(C(c3ccc(N(C)C)cc3F)=O)C2)C1 c1(N(CC(C)NC(c2cnc[nH]2)=O)C)nc(Cl)ncc1C(N)=O C1(CNC(c2onc(CCOCC)n2)=O)CCCN(C(=O)CSC(C)C)CC1 C1(C(=O)NC(C)(CNC(c2c[nH]nc2[N+](=O)[O-])=O)C2CC2)CCC(=C(F)F)CC1 CC1(C#CC(=O)N2CCCC(NC(c3ccccc3-n3ccnn3)=O)C2)CC1 c1(C(=O)NCC2CCN(C(c3n(CC)ncc3Cl)=O)CC2)c(C)nc(C)nc1C Cc1cc(C(=O)NCCCCN(C(=O)Cc2csc(C3CC3)n2)C)cc(F)c1C c1(CNC(=O)Nc2cc(C(=O)OC)ncc2)c(C)n(C)c2ccccc12 c1(OC(C)C(=O)NC2(CNC(=O)C(F)(F)Nc3cnn(C)c3)CC2)ccccc1 c1(OC)cc(Cl)c(NC(C2(C)CCN(C(c3cccc(F)c3Cl)=O)C2)=O)c(Cl)c1 C1(OCCC#C)CCN(C(=O)C(C2CC2)NC)C1 S(=O)(=O)(CCC(=O)NC)NCCN(C(=O)C(COC(C)C)NC(C)=O)C Cc1cc(=NC(=O)C2CCCC(NC(=O)C(C)(F)c3ccon3)C2)[nH]n1CCO C=CCC(C(=O)N1CC(OCC(=O)NCCc2cnc[nH]2)C1)C(C)C C1(NC(=O)NCCCNS(=O)(=O)c2ccccc2)CCCN2CCCCC12 c1(C(=O)NC(C2CCCC2)CNC(C(C)CCO)=O)cc2cc(Cl)ccn2n1 c1(-c2ccc(N3CCN(C(C=C(CCC)C)=O)CC3)cc2)cc(F)ccc1C CC1COCCN(C(=O)C(c2cccs2)NC(c2ncc[nH]2)=O)C1 CC1CN2CCN1CC2C(=O)NC1(CCNC(C2CCS(=O)(=O)C2(C)C)=O)CC1 CC1(C)C2CCC(C2)C1C(=O)NCC1(F)CN(C(=O)Cc2ccon2)C1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)N1CCCC(C(C)NC(c2ocnc2C(F)F)=O)C1 CC1(C(=O)NC(CC2CCCC2)C(=O)NC2C3COCC23)COCCO1 C(=O)(C1=CC2(CCOCC2)C1)N(C1CCCN(C(=O)C=Cc2cnc[nH]2)C1)C c1(C(N2CC(C(C)C)C(NC(C3(F)CC3)=O)CC2)=O)ccc2nccnc2c1 CS(=O)(=O)C1(C(N2CCN(C3CN(C(c4cnc(O)s4)=O)C3)CC2)=O)CCC1 C1(C)(CCC=C)CC(NC(=O)CCC(=C)Br)CN1C(C1CCOCC1)=O N1(C(C(C(CC)O)(C)C)=O)CCc2nc(CNC(c3cc(Cl)c[nH]3)=O)sc2C1 c1(C(=O)NCC2(C(N(CC)Cc3cccnc3)=O)CCC2)cc(N)cc(F)c1 c1(C(CC(=O)OCC)NCCC(C2CCOCC2)O)ccc(F)cc1 CC1CCN(C(c2cnc(Cl)c(C3CC3)c2)=O)CCN1C(c1cnnc(O)c1)=O CCC(CC(=O)NC1C2CCC1CN(C(=O)CNC(N)=O)C2)C(C)(C)C C1(C(=O)NC2C(CC(=O)Nc3cccc(CC)c3)CCCC2)C2CC3C(C2=O)C13 C1(COC)(CNC(C2CCCSC2)=O)CCCN1C(=O)CC1(C)CC1 C1(CNC(C2CC=C(C)CC2)=O)CC2(CO1)CN(C(=O)C(C)N(C)C)C2 C1(C(N(CC(C)OC)C)=O)(CNC(C2CCCS2)=O)CC(C)(C)C1 C1(C(N(c2nnc(CCC)s2)C)=O)CC(C)C(C(=O)OC)O1 CCCCS(=O)(=O)CC(=O)N(C)CC1(O)CCN(C(=O)C2=C(C)CCCC2)C1 C(=O)(C(C)CO)N(CCNC(C(=O)NC(C)C)=O)CCc1ccccc1 C(=O)(C1OCCc2ccccc21)NC(C1CN(C(CC=CC)=O)C1)C N1(C(c2ccc(C)cc2)=O)CC(CNC(c2coc(C(C)C)n2)=O)CC1(C)C c1(CN(C2CN(C(=O)OC(C)(C)C)C2C2CC2)C)cccc(Br)c1 C1(C2CCN(C(C3(Cl)CC3)=O)C2)(NC(C(c2c(OC)cccc2)OC)=O)CC1 C(=O)(C1=NN(C)C(=O)CC1)NCC(C)CN(C)C(C12CC(C1)S(=O)(=O)C2)=O C(C1CCS(=O)(=O)c2ccccc21)NC(N(C1CCCC(C)C1)CC(C)C)=O C1(C(N2CC3CCC(C2)N3C(C2(C(F)F)CC2)=O)=O)CCc2nncn2C1 CCC(CNC(c1sncc1C)=O)(CC)C(=O)NC1CC2CCCCN2C1 N1(C(c2n(C)c(O)nc2)=O)CCC2(CC1)CN(C(C1(C)CCCO1)=O)CC2CO C1(C(N(CCCNC(C2(c3cccc(Cl)c3)CCC2)=O)CC)=O)CC2C=CC1C2 c1(CC(=O)NC2OCC(CNC(=O)Cc3nnc(O)s3)C2)ccc(OC(F)F)cc1 N1(C(=O)Nc2cnc3scc(C)n32)CCCC(C2CN(C(=O)C3CC3)C2)C1 C#Cc1cccc(SCc2ccc(OCCn3nc(C)c(Br)c3C)cc2)c1C C(=O)(CC(O)CC(C)C)N1CC(C=C)C(NC(c2c(C)nsc2C)=O)C1 C1(C(N(CCNC(C(CC)C2CCOCC2)=O)CC)=O)C(C)OC(C)C1C c1(C(=O)NCCC(C)(C)NC(c2cc(OC)n[nH]2)=O)cc(Cl)c(Br)cn1 c1(C(=O)NCCNC(C(F)(F)C2(OC)CCC2)=O)ccc(=NCCOC)[nH]c1 C=C(C)CC(C)C(=O)NCCNC(=O)C(c1cccn1C)=O N1(C(C(C(CC)O)C)=O)CC2CCC(NC(=O)CC3CN4CCN3CC4)CC2C1 N(C(=NCc1csc(Cl)c1)NCc1cccnn1)C1C(C(F)(C#N)C2CC2)C1 C1(NC(C(C(=C)C)(C)C)=O)CC1C1CCCN(C(c2cccc([N+](=O)[O-])c2)=O)C1 c1(C(N2CC(NC(c3cccc(CC)n3)=O)C3C2C3)=O)ccc(C)cc1O c1(C(=O)OC)ccn2[nH]c(=NC(=O)CCc3cn[nH]c3)nc2c1 C1(C(=O)NC(C)Cc2cnn(C)c2)CCCCC1NC(C1CCC(F)C1)=O c1(SCC(=O)NC2CCC(N(C)C(c3ccn(C)c3)=O)C2)ccc(F)cc1 c1(C(N2CC(NC(C34CCOC3CCOC4)=O)C2)=O)cc(Br)cc(F)c1F Cc1nc2c([nH]1)C(C(=O)N1CCC3C(C1)CN3C(=O)COCC(F)F)CCC2 C(C(C)CC(=O)NC1CCCC1(C)NC(c1cc(C)n(C)n1)=O)OC N1(C(CC=C)=O)CCCC2(CCCN2C(=O)C(C2CCCCCCC2)O)C1 CCC(F)(F)C(=O)NC(CNC(c1ccc(CCC(N)=O)cc1)=O)CO c1(NCCCCNC(c2n(C)c([N+](=O)[O-])cc2)=O)nc(O)n(C)c(=O)c1[N+](=O)[O-] c1(C(=O)NCC2N(C(C3CCC(C)(C)O3)=O)CC2)c(Cl)cccc1[N+](=O)[O-] Cc1cc(N)c(C(N2CC(CNC(=O)CCCN3CCCC3)CC2C)=O)cc1C c1(OCC)nc(C)ccc1C(N1CCCC(NC(=O)COc2cnn(C)c2)C1)=O c1(CN2CC3N(C(c4cnc(Cl)c(I)c4)=O)C3C2)cc(Br)c(F)cc1F N1(CCNC(=O)OC(C)(C)C)CCCN(C(C2(C#N)CC2C(F)(F)F)=O)CC1 C=CCC(CC(=O)N1CC2CC2(C(=O)OC)C1)NC(c1cccc(CC)c1)=O N1(C(Cc2cccc(SCC)c2)=O)CCC2(CCN(C(=O)Cc3nccs3)C2)C1 N1(C(c2cc(OC)n[nH]2)=O)CCOC2(CCN(C(c3[nH]ncc3C#N)=O)C2)C1 Cn1ccc2cc(C(N3CCOC4CN(Cc5cc[nH]n5)CC34)=O)ccc12 C(=O)(C1=C(C)CCC1)N1CC(SC)C(NC(C2(C(C)C)CC2)=O)C1 C(=O)(C(C(=O)N(CC(C)CNC(=O)C=C(C)c1cnn(C)c1)C)C(C)C)OCC CC1CCOC(C(=O)NC(C)C(C)NC(=O)CCc2nc(O)n[nH]2)C1 c1(C(N2CC(NC(C3CC=C(C)CC3)=O)C3(C2)CC3)=O)c(F)ccc(Br)c1F C1(NC(c2cc(C)c(C)s2)=O)CCC2CCN(C(=O)CC3COC(=O)C3)C1C2 C1(O)(C(N)=O)CCCN(C(C2CC(O)CN2C(C2CCCN2C(N)=O)=O)=O)C1 C1(NC(C2OCCN(C)C2)=O)CN(C(=O)Cc2ccc(F)cn2)CCC1F C(C(O)CC(=O)N(C)CC1(O)CN(C(=O)CCc2cccc(O)n2)C1)N(C)C C=CC(CCC)CC(=O)N1CCN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CC(C)C1 c1(CNC(=O)Nc2ccc(OC(C)C)nc2)c(N)cc(F)cc1F c1(CC)nc(C)ncc1C(=O)NC1CCCCC1NC(C1CC(C)CCO1)=O N1(C(C2N(C)C(=O)CC2)=O)CC2CCC1(CNC(=O)Cc1cncnc1)C2 C1(CNC(=O)Cc2ccco2)CC(NC(c2csc(F)c2)=O)C12CCC2 CC12CN(C(=O)COCc3ccccn3)CC1CN(C(c1cc(=O)cc[nH]1)=O)C2 C(=O)(C(C)S(C)(=O)=O)N1CCC(CCNC(c2c(Cl)cn(CCC)n2)=O)CC1 N1(C(CC(=O)NCC)=O)CC(NC(c2cn(C)nc2C2CC2)=O)CC1(C)CC C(c1cnn(C)c1)=CC(=O)NC1(CC=C)CN(C(=O)CC2CCCC(OC)C2)C1 N1(C(CNC(C(C)CC2CC2)=O)=O)CCN(C(=O)C=Cc2ccsc2)CC1 C(=O)(C1=CC2(CCN(C(=O)CC3CCCOC3)C2)C1)N1C(C(=O)OC)CC1C N1(CCNC(C(=O)N(C(C)CNC(C2CC(C(F)F)C2)=O)C)C)CCOCC1 c1(CC)nn[nH]c1C(=O)NCc1ocnc1C(N1CC(n2cnnc2)C1)=O C(C(=O)NCCCc1nncn1C)(C(C)(C)C)OC O=C(C(F)(F)C(F)(F)F)NC1C2CCC1CN(C(c1cncc3n[nH]cc13)=O)C2 N1(C(c2c(CC)scc2)=O)CC2COCC(C1)C2NC(=O)CC1CCCCCC1 c1(C(=O)NCC(c2ccccc2)NC(C2C(C)C2)=O)cc(C(F)(F)F)cc(N)c1 c1(C(=O)NC2C3CCC2N(C(C2CC4(C2)CC4F)=O)C3)cnn2ncccc12 C1(C(N2CC(CC=C)(C(=O)NCCc3ncc(C)o3)C2)=O)CCOC(CC)C1 c1(C(=O)Nc2cc(I)ccc2Cl)cnc2[nH]cc(C3=CCCC3)c2c1 C1(CC)C(NC(=O)C(C)OC)CCN1C(c1cnn(Cc2ccccc2)c1N)=O N1(C(C2OCC(C)(C)C2)=O)CCC2CN(C(C3(C(F)F)CC(F)(F)C3)=O)CC12 CC1CCc2onc(C(N3CC(NC(c4cc5cccn5c(O)n4)=O)C3)=O)c2C1 c1(OC)cc(F)c(Br)cc1C(=O)N(C1CCCCC1)CCO.C(CS(=O)(=O)O)N C1(C2CC2)(CNC(C(C)=CC)=O)CCN(c2cc(OC)nc(COC)n2)C1 Cc1cc(C(N2CC=CC(C(=O)NCC(C)CC3CCC3)C2)=O)nn1C c1(-c2nn(-c3cc(F)cc(F)c3)c(-c3ccccc3)n2)cccn2ccnc12 CC1CN(C(c2cc(F)n[nH]2)=O)CCN1C(=O)Cc1cccc(F)c1F Cc1cnccc1C(=O)NC1(C)CCN(C(=O)CCC(=O)c2ccc(N)cc2)C1 N1(C(=O)C=Cc2cccnc2)C(CNC(=O)C(F)(F)C(F)(F)F)CC2COCC12 CCC(CCCC(=O)NCCC1COC(C)(C)C1)NC(=O)C(COC)(CC)CC N1(C(C2(CC)CCCCC2)=O)CC(NC(c2ccc(N)cc2O)=O)C(C)(C)C1 N1(C(C2CN(C(C)=O)C2)=O)CC(C(N2CCC(F)(C#N)C2)=O)CC(C)(C)C1 C(=O)(CC(C)C(C)C)NCC(C)N(C(c1cn(C)nc1OC)=O)CC Cc1cc(=O)c(NC(C2CCC(NC(c3cc(Cl)n[nH]3)=O)C2)=O)c(C)[nH]1 C1(C(=O)NC(CNC(C2(CC(=O)OC)CC2)=O)CO)(OC)CCCC(C)(C)CC1 c1(CC)ccc(C(N2CC3CC3C2)=O)c2ccccc12 C12(NC(C(Cc3c(C)nc[nH]3)O)=O)CCC(CC1NC(=O)C1=CCCOC1)C2 CC(C(=O)N(C1CCN(C(C2CCN2S(C)(=O)=O)=O)C1)C)C(C)(C)O N1(C(Cc2c(C)ocn2)=O)CCCC(CNC(=O)C(F)n2ccnc2)CC1 C1(NC(c2ccc(C)s2)=O)CC(F)(F)CC1NC(C1CC1OC(C)(C)C)=O N1(C(c2c(C)cncc2)=O)CC2CC1CN2C(c1cc(C2CCC2)[nH]n1)=O N1(C(C2C=C(C)CS2)=O)CCOC(C(N2CCC(O)(CO)C2)=O)C1 c1(NC2(c3nnnn3C)C(CCOC)COCC2)ccc(N2CCCC2)c(C)c1 N#Cc1cn(Cc2ccccc2)[nH]c1=NC(=O)N1CCC2(CCSC2)CC1 C1(CC=C)(C(=O)N(CC(C)(CC)OC)C)CCCN1C(=O)C(C)N=[N+]=[N-] C1(O)(CN(C)C(c2cccc(N)c2)=O)CCN(C(=O)CC(C)(C)C2CC2)C1 N1(CC)CCCC(Oc2ccccc2-c2cc(N(C)C)ccn2)CC1 C(C)(C(C)(C)C(=O)NCC1OCCC1(C)C)NC(COCC#C)=O C1(C(N2CC(C(N3CCCC3c3cccnc3)=O)C2)=O)CCCCC1(F)F C1(C(C(C)C)NC(C2(CCC)CCC2)=O)CCN(C(=O)CC2(C)CC2)CC1 c1(C(N2CCCC2C2(NC(C3C(COC)C3)=O)CC2)=O)ccc([N+](=O)[O-])cn1 c1(CN=c2[nH]cc(CCNC(c3sccc3Cl)=O)s2)ccc2nc[nH]c2c1 C12(CCN(C(=O)CCNC(C)=O)CC1)C(=O)NCC2.C1(CC)(CC)CC1 C(=O)(C(C)(C)C(C)NC(c1cccc(F)c1F)=O)NC(c1ccnc(C)n1)C C(=O)(C(C(=O)N1CCC1C(=O)Nc1ccc(N2CCCC2)cc1)OC)OCC Cc1nc(C(=O)NCC2(O)CC(NC(C3CC3c3cc[nH]n3)=O)C2)cc(O)n1 N1(C(c2ncc[nH]c2=O)=O)CC(CNC(C2(c3cccnc3)CC2)=O)C(O)C1 C1(C(C)(C)O)(CNC(COCCC)=O)CN(C(=O)CCC2CCC(C)O2)C1 c1(CC)nc(=NC(C)C2CCCN(C(=O)C(C)(C)n3cnnn3)C2)s[nH]1 N1(C(C(CCC)=CCC)=O)CC(CNC(C2CCN2CC)=O)C(C)(C)C1 C(=O)(C(C)(C)C(O)C(C)C)NC(CN(C(c1cc(CC)on1)=O)C)CC CCCCC(CNC(c1ccnnc1O)=O)NC(=O)C(C)(F)F CC1CCC(N(C)C(c2occc2CNC(C2CCCN2C)=O)=O)C1 Cc1csc2c(C(=O)NCC3CCCN3C(=O)Cn3c(C)csc3=O)ncnc12 c1(CC(=O)NC(CNC(C2C(COC)(COC)C2)=O)C)cnccc1Cl c1(C(N2C(CNC(c3n(C)nc(C4CC4)c3)=O)CC(O)C2)=O)ccc(F)cc1N c1(C(=O)NCC2(NC(C(C)CO)=O)CCCC2)sc(C#N)cc1Cl c1(OC)ccccc1CC(=O)NCc1ccc(C(C)NC(=O)CCN(C)C)cc1 N1(C(c2cc(C)c(C)nc2)=O)CCC2CCN(C(c3cc(C(C)C)[nH]n3)=O)CC12 CCCC(C(=O)NC(C)CC(C)NC(=O)C(C)Oc1ccccn1)S(N)(=O)=O C1(NC(C2CCCCC2(F)F)=O)CCN(C(=O)CSC(F)F)CC(O)C1 c1(C(N2C(CN(C(=O)C(N)=O)C)CCC2)=O)cn(C)nc1C1CCOC1 C(=O)(C1CCc2ccccc21)NC(CCNC(COCC(C)(C)C)=O)(C)C S(=O)(=O)(C1CC(c2ccccc2)C1)N(c1c(N(C)C)cccc1)C S(=O)(=O)(c1ccc(C#N)c(NCc2ncnn2C)c1)N1CCC(S(C)(=O)=O)CC1 C=CC(CC)CC(=O)N1CCOC(CCNC(C2CCCS2)=O)C1 N1(C(c2cc(C)nnc2)=O)CC2CCC1CC2NC(=O)C(C)C(F)(F)F N1(C(c2cc(=N)[nH]cc2)=O)CCCCC(NC(=O)CC2CC(C(F)F)C2)CC1 C1(CCC)CN(C(=O)COC(=O)CO)CCN1C(C1CCN(CC(F)F)CC1)=O N1(C(C(CN(CC)CC)F)=O)CC(N(C(=O)Cc2csc(=N)[nH]2)C)C2(CC2)C1 C1(CC)C=CCN(N2CC(OC)CC3(CCOCC3)C2)C1 c1(N(c2ccc(CC)cc2)CC=C)nnc(CC2CCOC2)n1CC CC1C(NC(=O)CC2CN3CCC2CC3)CCCN1C(=O)CSCCN(C)C N1(C(c2cnn(C3CCC3)c2)=O)CCC2(CC1)CN(C(C1CCC1F)=O)C2 C(=O)(C1=CCCOCC1)N(C1CCCN(C(C(c2ccc(Cl)cc2)=O)=O)C1)CCF C1(CNC(C2CCCO2)=O)CCC2(CN(C(c3cnc(F)c(Cl)c3)=O)C2)O1 CC1CCCCCCN1C(C1(C(C)C)CCN(C(c2cnn(CCF)c2)=O)C1)=O C1(CC)CCCN(CC(=O)NC2C3CC2N(C(C2(C(F)(F)F)CCC2)=O)C3)C1 C1(NC(C2C(C(C)NC(c3cc(C)sc3N)=O)C2)=O)CCCC1N=[N+]=[N-] c1(C(=O)NC(CC2CN(C(CN3CCC(C)C3)=O)C2)C)cnc2[nH]c(O)nc2c1 c1(OC(C)C)ccc(C(N2CC(NC(=O)CC3CC3(Cl)Cl)C(C(F)F)C2)=O)nn1 C(=O)(CCC(C(C)C)NC(=O)CCC1CCCN1C)N1CCC(C(=O)OC)CC1 C1(C(=O)NCC(CC)O)CC=CCN1C(=O)C=Cc1cc[nH]n1 c1(C(N2C(CN(C(C(CC)OC)=O)C3CC3)CCC2)=O)ccc2c(c1)CCO2 O=C(CCC(F)(F)C(F)(F)F)N1CCCC(NC(C23CC(O)C2C3)=O)C1 C(=O)(C(C)(C)CC(F)(F)F)NC1CCC(N(C(=O)Cn2cccn2)C)CC1 c1(OC)cccc(NC(C2CCCN2C(c2ccnc(C)c2)=O)=O)c1 S(=O)(=O)(c1ccc2c(c1)CCCO2)N1CCC2(CC(C)OCC2)CC1 N1(C(c2ccn(C(C)C)n2)=O)CCCC(NC(=O)CCn2cccn2)C1C Cc1cc(C(N2CC(C(C)NC(=O)CC3CCC(=O)N3)C2)=O)c(C)n1C CCCC(C)(CCC)C(=O)NC1CN(C(=O)CSCC2CCCCO2)CC1C c1(C(=O)NC2C3CN(C(C4CC(OCC)C4)=O)CC32)nccn2cc(C)nc12 C1(C2CCN(C(C34CC3C4)=O)CC2)(NC(c2nncc(C)c2)=O)CCOCC1 N1(C(c2cn(CC)nc2C)=O)CCCC2(C1)CN(C(C1CC(C)(O)C1)=O)CCO2 c1(OC)cccc(-c2nc(CN3CC(C)(C)C3)n(CC3(C(F)(F)F)CC3)n2)c1 C1(C(=O)NCC(CN(CC(=O)NC(C)C)C)(C)C)=NC=NNC(c2cccs2)=C1 C1(CNC(C2C(C)(C)COC2)=O)CCC2CN(C(=O)Cc3cncnc3O)CC12 c1(CC(=O)NC2CCCC2CNC(C2CC(O)C(F)C2)=O)cccc(OCCF)n1 c1(N(CCC)CCNC(c2ccccc2-n2cccn2)=O)nccnc1C#N c1(C(N(CCNC(=O)CCN2CCC2)CC)=O)ccc(N)c2cnccc12 N1(C(C2(C)N(C)CCC2)=O)CCN(C(=O)C(C)(C)S(C)(=O)=O)CC(C)(F)C1 N1(C(C2CC2(F)Cl)=O)CCN2CCN(C(c3n[nH]c4ccncc34)=O)CC2C1 N1(C(C(C(C)C)CNC(=O)CCC2CCCCC2)=O)CC(=O)N(C)CC1C c1(C(N2C(C(=O)NC(CCC)(C)CC)CC(O)CC2)=O)cnc(C)c(C#N)c1 C(=O)(CCC(F)(F)C(F)F)N1CCCC(F)(CNC(C=CC=CC)=O)C1 c1(CN2CC(NC(c3cc(C)n(C)n3)=O)C(F)C2)cc(Cl)c(Cl)cc1F c1(C(=O)NCCCC2(NC(c3c(C)ccs3)=O)CC2)cc(C2CC2)nnc1O C1(C(N(CC#C)CCO)=O)COCCC1NC(c1cccnn1)=O N1(C(CC(C(=O)OC)C)=O)CCN2CCOCC2(CNC(c2cn(C)cn2)=O)C1 c1(C(N2CC(NC(CC(CC)CC)=O)C3(C2)CC3)=O)ccc(F)c(C)c1C N1(C(Cc2ccc(C)o2)=O)CCN(C)CC1C(=O)NCC(C)(O)C(C)C N1(C(c2cc(C(N)=O)no2)=O)C2CCCC1CN(C(=O)CC1CCSCC1)CC2 CC1CC(C(=O)NCCC(=O)OC(C)(C)C)CCN1C(=O)C1=CC(C)(C)C1 c1(C(N2CCC(C3(NC(C(CCC)OC)=O)CC3)C2)=O)ccc2cnccc2n1 Nc1ccc(Cl)nc1C(N1CCCCC1CNC(=O)C(C1CCOCC1)O)=O C1(CCNC(COC(CC)C)=O)CCN(C(c2ccc(CO)o2)=O)CCC1(F)F c1(C(=O)NCC2CN(C(CC(=C=C)C)=O)C(C)C2)cccc(C(C)(C)C)c1N C(C(C)(C)CC(=O)NC(C1CCN(C(=O)COCC(F)F)CC1)C)NC(C)=O C1(CNC(C(CC)(C)CC)=O)CCCC2(CN(C(=O)CCC3CCOC3)C2)O1 c1(C(N2CCC(CNC(C3CC3CF)=O)C2)=O)ccnc2c(Br)cccc12 N1(C(c2onc(CC)c2C)=O)CCC(NC(c2coc3c2COC3)=O)C1(C)C Cc1ncccc1CC(N1CCC1(C)C(=O)NCC(c1ccccc1)O)=O CC1(C)CN(C(=O)C#CC2CCCC2)CCC1C(=O)NCC1(C(C)(C)O)CC1 C1(C(=O)NCC2(F)CN(C(c3c(CC#N)ccs3)=O)C2)CCC(=O)N2CCCC12 C1(NC(c2ccc(O)s2)=O)CC(CO)C2CC12.C(=O)(C1CC1)NC=O n1(C2CN(C(C(Cc3ccc(Br)cc3)NC(C)=O)=O)C2)cnc2ccsc2c1=O c1(OCC)ccc(F)cc1C(N1CCC2(NC(=O)Cc3ccoc3C)CC2C1)=O N1(C(CCC#CC)=O)CCN(C(=O)Cn2nnc3ccccc23)C(C)C1C N1(C(c2ccnc(C)c2C)=O)CCC2(CCCN2C(c2ccc(C(N)=O)[nH]2)=O)C1 N1(C(=O)CC=C(Cl)Cl)CCCC2CC12C(=O)O c1(C(N2C(C(N3CC(C)OCC3)=O)CC(O)CC2)=O)cc(C2CC2)nc(Cl)c1 c1(C(N2CCC(C(=O)OCC)C2)=O)ccnc(O)c1F C1(C(=O)NC(CCCC)CNC(=O)CCF)CC2CCC(C1)S2 C(=O)(C1=CCCOC1)N(C)CC1CCC(CNC(C(CC)CC)=O)CC1 N1(C(C(C)O)=O)CC2CCN(C(c3csc(Cc4ccccc4)n3)=O)C2C1 CC(C)CC(C(=O)N(CC(O)CN(C(=O)C(C)SC(F)(F)F)C)C)C(N)=O c1(NC(C(C)C)CCNC(=O)CC2(N(C)C)CC2)ncccc1[N+](=O)[O-] N1(C(c2c(C)ccs2)=O)CCC2(CCCC2C(N2CCOC(C)(C)C2)=O)C1 CC(CCCCNC(c1csc(C#N)c1)=O)NC(=O)CC1C=NN(C)C1=O N1(C(c2cc(C#N)sc2)=O)CCC2(CC2)CC1C(N1CC(F)CC1CO)=O C(=O)(C1CCCc2nn[nH]c21)N(C(C)CCNC(C12CCCC(C)(C1)OC2)=O)C C1(OCC)(CNC(=O)CC2CCCN2C(=O)C(C)(F)F)CN(C)C1 c1(CC)cccc(F)c1C(=O)N(CCCNC(c1ccc(Br)nc1O)=O)C c1(NC(CC(C)N(C(C(COC)(C)OC)=O)C)=O)ccc(C)cc1OC c1(C2C(=O)C2C)cccc(OC(C)=O)c1.C1(CCN)CCCC(OC)C1.N(C1CC1)(CC)O C1(O)(CN(C)C(c2sccc2C#N)=O)CCN(C(c2n[nH]c(C(C)(C)C)n2)=O)C1 C(=O)(C1=CC2CCC1C2)N(CC(C)NC(c1ncccc1C(F)F)=O)C c1(CN2CC3N(C(c4ccc(C)nc4Br)=O)C3C2)c[nH]c2cccc(Cl)c12 N1(C(C2CCC(NC(C3N(C)CCC3)=O)C2)=O)CCC12CCSCC2 c1(C2CCCN(C(C(CC=C)(C)O)=O)C2)ncc2n1CCCC2 c1(CNC(N2CCCC(CCOC)C2)=O)ccc2c(c1)OC(C)(C)O2 C1(NC(c2c(SC)ccs2)=O)CC2COCC(C1)N2C(C1CC2C=CC1CC2)=O C1(CC)COC(C)(C)CN1C(=O)CCOCCNC(c1cc[nH]c1)=O C(C1CCCN1C)=CC(=O)NC(C)CC1CN(C(c2ccnnc2)=O)C1 c1(OCC)ccccc1C(=O)NCCCN(C(=O)C(O)COCC(F)(F)F)CC c1(C(N(C)Cc2ccccn2)=O)ccnc(CNS(C)(=O)=O)c1 N1(C(C2CCC(C)(C)O2)=O)CCC(O)C(NC(C2CCOCC2(C)C)=O)C1 C1(C(C)CNC(C2(C)CCCO2)=O)CCN(C(=O)C(F)OC(F)(F)F)CC1 N1(C(COC2C(CC)CCCC2)=O)CCC(CC)(NC(C2C=CCC2)=O)CC1 CC1=CCC(C(=O)NC(C)CC(=O)NCC(C)(C)C2CCC2)CC1 C1(NC(=O)COC2CCCC2)CCC2(CC1)CCN(C(=O)C(F)n1cccn1)C2 c1(CC(N2CC(N(C(CC(C)C)=O)C)C(F)C2)=O)cc(F)cc(Cl)c1 CCCCCC(C)CC(=O)Nc1nc(-c2cc(CO)ccc2F)cs1 CCCCC(C(=O)NC)NC(C1CN(C(=O)CC2(N(C)C)CCC2)CCN1C)=O c12cccc(c1)CN2C.C(=O)(C(=O)N(C)C(c1ccco1)C)NCC C1(O)(C(=O)NCC(=O)NC2CC2)CCCN(C(=O)CC(=O)NCc2nc[nH]n2)C1 CC1CCc2[nH]nc(C(=O)NC(C)Cc3cccc(Br)c3)c2C1 c1(C(N2CCC(CN(C(C(CC)OC)=O)C)CC2)=O)cnn2ccnc(N)c12 c1(SC)ccc(C(=O)NC2CN(C(c3nccn3C)=O)CC2F)cc1 C(=O)(C(C(=O)N(CCC(C)NC(c1cnn(C(C)(C)C)c1)=O)C)C(C)C)OCC N1(C(C=CC=CCCCCC)=O)CCCC(NC(=O)Cc2ncoc2C)C1CC c1(C(=O)NCC(C2CCOC2)NC(=O)Cn2cnnn2)cnc2c(c1)CCOC2 c1(NCCc2n(C(C)C)cnn2)cc(=NC2CCCCC2CO)[nH]c(C(C)C)n1 C1(C(C)NC(=O)CCCN2CCCC2)CCCN1C(=O)C(C)(C)C1CCCC1 C1(CNC(CCCOC(C)C)=O)CN(C(C2CCN2S(C)(=O)=O)=O)CCN1C CC(CN(C(=O)CN=S(C)(C)=O)C)N=c1nc[nH]s1 C1(C(c2ccccn2)C(=O)OCC)CCN(N2CCSC(C)C23CCC3)CC1 N1(C(CCSc2n(C)nnn2)=O)CC2CCC1CN2C(=O)CNC(=O)C(=O)O N1(C(C(C)C#N)=O)CC2CC(NC(C3CC4(CSC4)C3)=O)C(C2)C1 C1(CC=C)(NC(c2csc(C3CCCO3)n2)=O)CCN(C(=O)CCSCC(C)C)C1 c1(C(N(CC(=O)N(CC(C2CCC2)OC)C)C2CCC2)=O)cc(F)c[nH]1 c1(NC2C(C3CCN(C(C4(Cl)CC4)=O)CC3)OCCC2)ncnc(O)c1Br CCCC(CCc1ccccc1)C(=O)NCC(C)(C)NC(=O)C1=CC(O)CCC1 N1(C(C(c2ccn(C)c2)C)=O)CCC(F)(C(=O)NCCOCCN(C)C)C1 c1(C(C)NCCCCCOC)cc(Cl)ccc1OC(F)(F)F c1(C(N(C(C)CNC(C2(C)CCCCO2)=O)CC)=O)ccn2ccnc2n1 N1(C(c2ccc(CS(C)(=O)=O)cc2)=O)CCC2(CCN(c3snc(Cl)c3C#N)C2)C1 C1(CNC(c2nccc(SC)n2)=O)C(C)CCCN1C(=O)Cc1cc(C)cs1 c1(C(=O)NCCC(F)Cn2cc(C3(O)CC3)nn2)cc(Cl)nc(Cl)c1 c1(C(N2C(CNC(C=NOC)=O)C(C)CC2)=O)cc(Cl)c(F)c(Cl)c1 C(=O)(CCS(N)(=O)=O)NCC(C1CCCN(C(C2(CC)CCCCC2)=O)C1)(C)O CON(C)C1CCN(C(c2cnn(CCNC(c3nc(=N)cc[nH]3)=O)c2)=O)CC1 Cc1[nH]c(=NCC(C)(C2CC2)NC(C2CN(C)CC2C(F)(F)F)=O)ccc1C#N C1(C(C(=O)NCC2C(NC(c3cn(C4CC4)cn3)=O)C2)O)CCCCC1 C(CCCCC(=O)NCCCCC(CO)NC(=O)C(C(C)C)n1ccnc1)=CC c1(C(CC)C)ccccc1NCC1CCOCC1NC(=O)OC(C)(C)C Cc1nn(C)c(N)c1C(=O)NCC1CN(C(=O)CCC(=O)NC2CCCC2)CCO1 C(C(O)C(C)(C)CO)NC(C(N1CCC(N(C)C)CC1)=O)=O Cc1c(C(=O)NCC2CC3(CC3)CN2C(c2cccc(Cl)c2)=O)sc2nccn12 Cc1cccc(NC(=O)COC(N2CC(C)(Nc3cccc(COC)c3)C2)=O)n1 N12CCC3(CC3)CC1c1nc(no1)CC(N=[N+]=[N-])C2=O.C12CC3(CC13)C2=O.CO CCCCC(CCC)NC(=O)C(CNC(c1cc(F)cnc1O)=O)C(C)C C1(CC(=O)N(CCN(C(c2[nH]ccc2C2CC2)=O)CC)CC)CCCC(C)O1 c1(C(N2CC(CC)N(C(C3CN(C(C)=O)C3)=O)CC2)=O)ccc(S(C)=O)cc1 C1(C(N2CCC(O)(CCNC(c3sccc3F)=O)CC2)=O)CCC2CCC(=O)N12 N1(C(CC(CC)(C)C)=O)CCC2CN(C(C3CCC4(CC4)C3)=O)CC2CC1 N1(C(CCC=C=C)=O)CCC2(CCCN(C(c3sc(C4CC4)nc3C)=O)C2)C1 N1(CCNC(c2c(CC)nc[nH]2)=O)C(C)CCC1C N1(C(COCC(=C)C)=O)CCC(NC(c2cn(CCC)nn2)=O)C(CO)C1 C1(CC)(NC(=O)CS(N)(=O)=O)CCN(C(c2nc(C(C)C)cc(C)n2)=O)CC1 c1(C(=O)NCC2N(C(c3nc(C)oc3)=O)CCC2)cnc(CC2CC2)nc1O CC(C)C(C(=O)N1CCCC1(C)C(=O)Nc1ncc(Cl)s1)c1ccc(F)cc1 n1(CC(=O)N(C2CCCN(CCn3cncn3)C2)C)ccc2ccccc12 N1(C(=O)CCCCBr)CCC2(CC1)CCN(C(c1ccc(C(F)F)cn1)=O)CC2 Cc1cc(F)c(C#N)cc1NC(C1CC(NC(=O)CCn2cncn2)C1)=O C1(C(=O)NC2CCN(C(c3c(Cl)n[nH]c3C3CC3)=O)C2)CC2CC1CC2(F)F c1(C(=O)NCCC23CN(C(CCCCCC)=O)C(CC2)C3)snc2ccccc12 c1(CC)cc(F)c(C(=O)NC23CCC2CN(C(C2NC(=O)OC2C)=O)C3)cc1F C(=O)(C(=O)N=S(C)(C)=O)NC(C1CCCN1C(=O)Cn1nccn1)C C(=O)(CCCCCC#N)NCC1N(C(C(C)(F)F)=O)CC(F)C1 c1(C(C)(C)C)nc(=NCC(F)C2(c3ccccc3)CC2)s[nH]1 C12(CNC(C(CC#C)C)=O)CCC(CC1)N2C(c1c(Cl)cccc1Br)=O N1(C(c2nc(CCC)oc2)=O)CC2CC(NC(=O)CC3(CSC)CC3)CC2C1 c1(CC(=O)NCC2N(C(c3c(C)con3)=O)CC2)c(C)ncnc1C C(c1ccccc1C)=CC(=O)NC1CC(N(C(c2c(CCC)nco2)=O)C)C1 c1(NC(NC(C2CCCCO2)CC)=NC)ccc(N2CCC(C)CC2)cc1 Cn1nccc1C=CC(=O)NC1CCCN(C(=O)C(F)(F)CF)C1 C(CC(N)=O)(C(=O)N1CCN(C(=O)CC2CCCCC2)CC1)NC(CC(C)C)=O N1(C(c2c(C3CC3)[nH]c(=N)s2)=O)CC2CCC(C1)C2N(C12CCCCC1C2)CC CCCCCC(O)CC(=O)NC1CN(C(c2cc(F)ccc2C)=O)CC1C C1(C(=O)NC(CCOC)CNC(=O)C2=CCCS2)CSc2ccccc2O1 c1(C(=O)NC2(C)CCN(C(c3c(CC)n(C)nn3)=O)C2)n[nH]c2ccc(C)cc12 c1(SCC(=O)NC2CC(CNC(C(=O)NCC)=O)C2)nnnn1C CCCCCCC(F)C(=O)NC(CCNC(c1cnc2n1CCOC2)=O)C(C)C N1(C(c2ccc(SCC)nc2)=O)CCOCC(C)(CNC(C2CC=CCO2)=O)C1 C1(C(=O)NCC(CNC(c2cc(-n3cccn3)on2)=O)O)CCN(C2CC2)CC1 CCC(CCCC(=O)NCCC(C)CCO)NC(=O)C(COC)COC C1(CNC(C2CC2(Cl)Cl)=O)CCC2(CN(C(=O)CCc3cncnc3)C2)O1 N1(C(C(CN(C)C)N(C)C)=O)CCCCC(NC(C2CC(N(C)C)C2)=O)C1 c1(N2CC(SC)CC23CCC3)ccc(S(=O)(=O)NCCCN2CCOC2=O)cn1 N1(C(n2ncc(C#N)c2)=O)CCC(C2CC(NC(C3(N4CCC4)CCC3)=O)C2)C1 C(CC(C)C)(C(=O)NCC(c1ccccc1)NC(=O)C(=O)NC(C)C)OC C(C)(C(=O)COC(C1(O)CCSC1)=O)OC N1(C(C(=O)N(CC(F)Br)C)=O)CCc2nc(C(F)(F)F)ncc2C1 C1(CNC(C(CCC)(C)CC)=O)Cc2ccccc2CN1C(=O)CN(C)C1CC1 c1(CCC)cc(C(=O)N(CC(CC)NC(C2CC(C#N)C2)=O)CC)no1 C1(NC(C(C)NC(C2(CC)COC2)=O)=O)CCCSC1 c1(CN(c2ccco2)Cc2cc(OC)cc(Cl)c2)ccc(C)c(C)c1C N(S(=O)(=O)N1CC2CCC1C2)CC(N1CCCN(CC)CC1)=O c1(C(=O)OC)ccc(C)nc1NC(C1(C)CCCN(Cc2cc(C)ccn2)C1)=O N1(CCNC(C(CC)CC)=O)CCCN(C(C2(c3ccc(Cl)cc3)CC2)=O)CC1 C1(C(=O)NC2CC(C)(NC(C3CC4COCC4C3)=O)C2)CCC2(CCC2)CO1 C1(F)(C(C)C)CCN(C(=O)C(C)(C)NC(=O)CCCOc2ccccc2Cl)C1 C1(C(=O)NC(C)CNC(=O)CCC(=O)c2ccc(Br)cc2)CCc2c[nH]nc2C1 N1(C(CCOCC)=O)CC2CC1CN(C(=O)C(C)C(F)(F)Cl)C2 c1(C(N2CCC(C(=O)Nc3ccc4nn[nH]c4c3)C2)=O)cccc(O)c1[N+](=O)[O-] c1(CC(=O)NCCNC(C2(COC)COC2)=O)ccc(C(F)F)cc1 c1(C(N2CCC(N(C(c3cc(C)oc3)=O)C)C(C)C2)=O)cc(N)c(Cl)c(O)c1 C1(C(N(C2CCN(C(c3cnn(C)n3)=O)C2)CCO)=O)CN2CCC1CC2 Nc1c(C(N2CCN(C(c3cccc4ncnn34)=O)C3CC23)=O)cc(F)cc1Cl Cc1csc(C)c1C(=O)NC(CC(=O)NC(c1ccc(O)nc1)C)C1CC1 C(C)(C)(CC(F)C(=O)N1CCC(C(C)(C)O)CC1)NC(C(C)N(C)C)=O c1(OC)cc(C2CC2C(=O)NCC2(OCCO)CCSC2)ccc1F c1(C(C)C)nc(NCCC2CCC(C)O2)cc(=NC(C)c2ccc(F)c(F)c2)[nH]1 c1(C(N(C2CN(C(=O)C3=NOCC3)CC2F)C)=O)ccnc(O)c1Br c1(C(=O)NCC(CC)NC(=O)C(C2CCS(=O)(=O)CC2)O)c(C)cccc1N CC(C)C(C(=O)NCCN1CCNC(=O)C1)NC(=O)Cc1cc[nH]n1 N1(C(CCC(=O)NCCNC(C)=O)=O)CCC2CN(C(=O)CC(C)C(C)(C)C)CC12 c1(C(=O)NC(C(C)NC(C(COC)C)=O)(C)C)cc2c(Br)cccc2c(O)n1 C(=O)(C1CCc2cccnc21)NCC1(O)CN(C(C2CCCC(=O)CC2)=O)C1 C(=O)(C(O)CCCCC)NCC(C1CC1)NC(CCC(=C)Br)=O C(CCCC(=O)NC1(CCCNC(=O)C(C)(C)N2CCCCC2)CC1)N(C)C C1(NCc2cccc(C=C)c2)CCC2(C1)CN(C(=O)CCc1ccccn1)C2 C(=O)(C1=CCCSC1)NC1CC(CNC(c2c(C)onc2C2CC2)=O)OCC1 N1(C(C=CCOCCOC)=O)CCC2(CC1)CC2CNC(=O)CNS(N)(=O)=O N1(C(CC(C)SC)=O)CCCC(NC(=O)CCc2ccco2)C1 CCC(C)(C(=O)NCC1CN(C(c2n[nH]c3c2CCSC3)=O)CC1C)C(N)=O c1(N2CC3(C(C(=O)NCC4(C#N)CC4)C3)C2)ncnc2c(Br)c[nH]c12 C1(C(N(CCOC2CCN(C(C(C(C)C)C)=O)CC2)CC)=O)CCCCC1(F)F c1(COC)nn[nH]c1C(=O)NCC=CCNC(=O)CCn1cccn1 C1(C(C)C)CCN(CC(=O)NC(c2cccc(Cl)c2)C)CC1 c1(N2CCC(=CCNC(c3nncc(OC)c3)=O)CC2)nc(Cl)ncc1Br c1(N(C2CCOCC2)C(c2ccc(Cl)cc2)(C(C)(C)OC)C)ccc(OC)nc1 c1(C(=O)NCC2C(C)CCN(C(=O)C3=CCC3)C2)cccc2c1COCCN2 N1(CC(=O)NCC(C)(C2CC2)SC)CC2C(C(=O)NCC(=O)OC(C)(C)C)C2C1 C(=O)(CC(C)(C)CC(F)F)N1CC(NC(CSc2n(C)cnn2)=O)C2C(C1)C2 C(=O)(CCC1=NNC(=O)CC1)NC1C2CCN(C(c3c[nH]c(=N)s3)=O)C2C1 C1(C(=O)NC2CCCC(CNC(c3cnn(C)c3Cl)=O)C2)COC2(CCC2)CO1 C1(NC(C=C=C(C)C)=O)CN(C(c2cc(C)nc(C)c2O)=O)C2CCCC12 c1(C(=O)NC(C2CCN(C(c3coc(C(F)(F)F)c3)=O)C2)C)cccnn1 N1(C(C(CCCC)NC(N)=O)=O)CCC(F)(F)C(CNC(c2conc2C)=O)C1 c1(C(=O)NC(C(C)(C)O)C(=O)O)ccc2c(c1)nc(O)n2C1CC1 N1(C(COCC(C)C)=O)CCC2(NC(c3cc(=O)n(C)cn3)=O)CCCCC12 C1(CC(=O)NCC(CNC(C=CC)=O)(C)OC)CCOCC1(C)C C1(NC(C2N(CC)CC2)=O)CCN(C(=O)C(C)(C)CC2CCOCC2)CC1 C1(C(N2CC(N(C(c3cc(CCC)n(C)n3)=O)C)C2)=O)CS(=O)(=O)CCO1 CC1(C)CC2(CC2C(N2CCOCC2CNC(=O)COc2cccc(Cl)c2)=O)C1 Cc1ccc(C(=O)NC2CN(C(c3ccc(F)c(F)c3)=O)CC2C)c(O)c1 Cc1cc2cc(C(=O)NCC3CCCN(C(C4CCOC4)=O)CC3)[nH]c2cc1Cl C(=O)(C(C)CNC(=O)Cc1cc[nH]c1)NC(c1cccs1)CC c1(CC(=O)NCC(c2ccccc2)NC(CCOCCC)=O)ccn(C(F)F)n1 CC(C(C)(C)NC(=O)CCc1ccsc1)NC(c1c[nH]nc1C(F)F)=O c1(CC(C(=O)NC(COCC)C(C)C)C)ccc(F)cc1F C1(NC(=O)COC2CCCCC2)CCN(c2nnnn2-c2ccccc2)CC1O Cc1cc(C#N)ccc1C(N1CCC2CCCC12C(=O)NCC(C)O)=O n1(CCC(=O)NC2CC(C)(NC(CC(CCC)O)=O)C2)cc([N+](=O)[O-])nc1C C=C(C)CCCC(=O)NC(C1CCN(C(=O)Cc2cc[nH]c2)C1)C c1(CC)ccc(C(=O)NC2CC2NC(C2CCCCN2C(C)C)=O)c(F)c1 c1(C(N(C2CCC(NC(CC)=O)CC2)CC)=O)n[nH]c2cc(C)ccc12 C1(NC(CCCC#CC)=O)COC2(C1)CN(C(c1ccc(C#N)cc1)=O)C2 N1(C(C2(CC=C)CCOC2)=O)CCN(C2CN(C(=O)C(F)=CC)C2)CC1 N1(C(c2c(C)ncc(N)c2)=O)CCC(NC(C2CCC2(F)F)=O)CC(C)(C)C1 C(=O)(C(C)(F)CCCC)N1CC(O)(C(C)NC(C=C(CCC)C)=O)C1 C1(CC(NOC(CC)CC)=O)N(C(=O)COCC2CC2)CCC1(C)C c1(CC(N2CCCC(N(C(Cc3cc(C)on3)=O)C)C2)=O)csc2nccn12 N1(C(c2ccc(CC)[nH]2)=O)CC2CS(=O)(=O)CC2(NC(c2ccnnc2O)=O)C1 C(=O)(CCCC(CC)NC(c1cnc(O)c(C)c1)=O)NCc1ccc(CC)cn1 CC(CC(C)(F)F)C(=O)NC1CCC(NC(=O)CC23CCCCC2C3(F)F)CC1 C=CC(CCC)CC(=O)N1CCC(C)C1C(N1CCCC(C)(C)C1)=O CCCCCCC(=O)N1CCOCCC1C(=O)N(C)Cc1nc(CC)no1 c1(C(N(CC(CC)NC(=O)C(C)NC(C)=O)C)=O)ccc(CN(C)C)o1 N#Cc1cccc(OC(c2cccc(N3CCCC3=O)c2)=O)c1 N1(C(c2ccc(SC)s2)=O)CC(NC(C2CCCC(CF)C2)=O)C2(CC2)C1 C1(NC(c2c(C)nsc2)=O)CC(CNC(C23CC(C)(CCO2)C3)=O)C12CCC2 C(C)(C)(CC(C)NC(c1cc(CNC(c2coc(C(N)=O)c2)=O)[nH]n1)=O)OC N1(C(CSC)=O)CC(NC(c2nnn(-c3cc(C)ccc3C)c2C)=O)C(C)(C)C1 C(CCC(=O)N(CCSC)CC)(C(C)C)NC(CC(CC)OC)=O C12(C(N(CCCCC(=O)NCC(C3CCC3)OC)C)=O)CCCC(CO1)C2 C(=O)(C1CCCc2nccn21)NC12CC(NC(CN(S(N(C)C)(=O)=O)C)=O)(C1)C2 c1(C(=O)NC2CCCN(S(C(CC)C)(=O)=O)C2)ccc(Cl)c(Cl)c1 N1(C(C(C=C)O)=O)CCCC1(C)CCC(=O)NCc1cc(O)ns1 Cn1cnc(I)c1C(C(=O)NCC1CCOC1)N1CCC1c1cccnc1 c1(C(=O)NCc2ccc(-c3cncc(C#N)c3)cn2)cn2ccccc2n1 Cc1ncc(Cl)c(C(=O)NC2CCCCC2NC(=O)CCOCC2CCCO2)n1 C1(O)(CN(C(c2cc(CC3CC3)on2)=O)CC)CCN(C(=O)C(C(C)O)N(C)C)C1 C(CN=c1[nH]c(C(=O)N(C)C)cs1)c1scc(C)c1 c1(CN2CCN(C(C3CCCN3)=O)CC2)cc2cc(Br)cc(F)c2o1 C1(OCC(N)=O)CCN(C(C2OCCC2NC(=O)Cn2ccnc2)=O)C1 N1(C(c2c(CC)n(C)nn2)=O)CCC(C(=O)NC(C)CCOC)C(C)C1 C1(C(=O)NCCC(Cn2cc(CCCOC)nn2)F)CCc2c(cnn2C)C1 C1(CNC(C2CN(C)C(=O)N2)=O)CC2(CO1)CN(C(c1ccoc1)=O)C2 N1(C(Cn2cc(C(C)NCC)nn2)=O)CC(C)=C(C)C1 n12cc(nn1)CNC(C)C2.c1(C(=O)OCCCCO)csc(CO)n1 CCC(CC)C(F)C(=O)NCc1ccc(C(=O)NCC(C)C(=O)OC)cn1 C1(CC(=O)NCC2CCN(CCC)C2)CCCCN1C(c1cnn(C)c1CC)=O C1(CCNC(CN(C)C(=O)C2CC2)=O)CCCCN1C(c1[nH]ncc1C#N)=O Cc1cc(C(N2CCC3CC23C(=O)NCCN(C)C)=O)cc(O)n1 c1(C(=O)NCCN(C)C(c2nnn3c2CCC3)=O)ccc2cnoc2c1 c1(C(N2CC(F)(C(N3CC(OC)OCC3)=O)C2)=O)ccc(Br)c(C)c1F c1(C(=O)NC2(CO)CN(C(C(CCC)OC)=O)C2)ccnc(O)c1Br C1(CNC(c2cc(SC)oc2)=O)C2CN(C(=O)C(C)(c3cccs3)N(C)C)CC12 Cc1ccccc1S(=O)(=O)CC(=O)NCC1CCN(C(c2ccns2)=O)CC1C N1(C(CC=C)=O)CCC2(CC(C(=O)NCc3c[nH]nc3C(C)C)=NO2)C1 C1(CNC(C(c2ccccc2Cl)OC)=O)COCCN1C(c1c[nH]ccc1=O)=O n1(Cc2onc(C(C)SCC)n2)c(-n2nc(C)cc2C)nnc1C1CCCC1 N1(C(C(CCCOC)C)=O)CCc2ccc(C(=O)NC(C)C)nc2C1 C(=O)(CC(C)(O)C(F)(F)F)N1C2C(NC(c3c(OC)cncc3)=O)CC(C2)C1 N1(C(CC(C)OC)=O)CCCC(NC(=O)CC2(C(F)(F)F)CCC2)C1 Nc1cc(C(=O)NC(CCF)C(=O)NCc2cncs2)cc(F)c1 c1(C(N(CCOC)CCNC(c2c[nH]nc2C=O)=O)=O)cc2cccc(F)c2o1 CC1(CNC(=O)C2=CCSC2)CCCN(C(c2ccc(F)cc2Br)=O)C1 N1(C(C2CC(C)(NC(C(CSC)O)=O)C2)=O)CCC(F)(CO)CC1 c1(C(C(=O)NC2C(NC(Cc3cc(COC)on3)=O)COC2)(C)C)cccc(F)c1 c1(C(N(CC(C)NC(C(C(=O)OCC)CC)=O)C)=O)cc(S(C)(=O)=O)c(C)o1 CC1CN(C(c2sccc2C2CC2)=O)CCCN1C(c1ccnc(Cl)c1N)=O c1(C(N2CC(NC(CCOC(C)C)=O)C(CO)CC2)=O)ccc(=O)n2c1CCC2 c1(C(CC(=O)NCC(CC)NC(C2(C)CCN(C)C2=O)=O)C)ccc(F)cc1F c1(C(N2CCC(C(C(=O)NC3(c4cccs4)CC3)F)C2)=O)cccn2ccnc12 c1(CC)ccc(Cl)c(S(=O)(=O)N2CCCC2c2ccc(O)cc2)c1 CC1CC(NC(c2cnn(-c3nccs3)c2)=O)CN(C(=O)CC2CCCN2C)C1 C(=O)(CS(=O)(=O)C(C)(C)C)N1CCC(C2(NC(c3n(C)c(=O)ccc3)=O)CC2)C1 c1(C(=O)NCC(CC=C)NC(c2cc3cccnc3[nH]2)=O)ccc2nncn2c1 c1(C(=O)NCC(C2CC2)NC(C(CC)OC2CCCC2)=O)cc(N)cc(O)n1 Cc1cc(C)c(C(=O)NCCC2CCN(C(c3n[nH]c(C)c3C)=O)C2)[nH]1 N1(C(c2c(C)ncnc2)=O)Cc2n[nH]cc2C1C(=O)NCCC(O)C(F)(F)F Cc1cc(C(=O)NC2CC(N(C(=O)C3=CS(=O)CCC3)C)C2)cn(C)c1=O C12(C(=O)OC)CCCOC1CN(C(=O)Cc1ccncc1Cl)C2 c1(-c2c(C(=O)OC)ccc(Cl)n2)ccc(N(CCNC)CC2CC2)c(C)c1 c1(C(=O)NCC(C)(CC(C)C)NC(c2c(C)cco2)=O)ccc2c(c1)OCO2 C(=O)(C(C)CS(C)=O)N(CCN(C(C)C)C(c1ccn(CCN(C)C)n1)=O)C C1(C(=O)N(C2C(C(C)NC(=O)COC3CCC3)C2)CCO)CC2CCC1O2 CC1CCCN1CC(=O)N(C)CCOCCNC(C1(C(F)F)CC(O)C1)=O Cc1cc(C(=O)NC(C2(O)CN(C(=O)C(C)Sc3ccccc3)C2)C)ccn1 C(=O)(C(C)(C)C(C)C)NC(C(C)C)CNC(=O)CC1(C)CC1(F)Cl N1(C(C2C(C)C2)=O)CC(NC(c2nn(C)c3c2CCCC3)=O)CC12CCOCC2 C1(C)(CNC(C2CC(CCC)C2)=O)COCCN(C(c2cnn(CCF)c2)=O)C1 c1(OCC)ccc(NC(N2CCCC2(C)c2cn(CC3CCCO3)nn2)=O)cc1 C(=O)(C(O)C(C)c1ccccc1F)OCCN(C(C1CCN(CC)C1)=O)CCF c1(C(=O)NCCN(C(CCSC)=O)CC2CC2)cnoc1-c1ccc(Cl)s1 C(=O)(C(C)(C)CCCO)NC1CN(C(c2cc(CC)[nH]n2)=O)C(C)CC1 Cc1cc(F)ncc1C(=O)NCCC(C)N(C)C(c1cc(C(F)(F)F)cs1)=O c1(CNC(C(CC)OC)=O)cccc2c1CCN(C(=O)C(CC)C(=O)OC)C2 S(=O)(=O)(c1c[nH]ccc1=NC1CCCCCCC1)N.O=C1NC(=O)C2(CCCC2c2ccccc2)N1 N1(C(CCCOCCC)=O)CCN(C(c2cccc(O)n2)=O)C(CC(F)(F)F)C1 C(CN(C)C)(N=c1ccnc(N(C)CC2CC2(F)F)[nH]1)c1c(OC)cccc1 CC(C)CCCC(C)C(=O)NC1CC(C(N2CCOCC23CC3)=O)C1 CCCC(C#N)C(=O)N1CCC1CNC(c1cc(C(C)(C)C)no1)=O Cc1cc2ccc(C(=O)NCC(C)(O)CNC(c3nc(C4CC4)cs3)=O)cn2c1 C1(CNC(c2ccc(SC)o2)=O)CCN(C(c2cc3n(n2)CCO3)=O)CC1C c1(OC)cc(OC)nc(C(=O)NC(C)CCNC(C2CCCCC2C)=O)n1 C1(NC(C(CC(=C)C)NC(c2ccnc(C)c2N)=O)=O)CCn2cncc2C1 Cc1ncc(C(F)(F)F)cc1C(=O)NC(C)CC(C)NC(=O)C1=CCCOC1 CCC(CCCO)NC(=O)CCNC(C1(CC)CCCC1)=O c1(C(=O)NCC(CNC(C(C)Cn2cccn2)=O)O)cc(Cl)cnc1O C1(NC(C(=O)NC(C)CN2CCOCC2)=O)CCCC2CNCC12 N1(C(c2c(Cl)cn(C)n2)=O)CCCCC(CNC(=O)CCCN2CCOC2=O)C1 CC#CCC(CO)NC(C1CCN(c2ccccc2F)C1)=O C(=O)(C(C)S(C)(=O)=O)N1C(CC)C(C(=O)NCc2ncnn2C(C)C)CC1 C1(C)(NC(C2CCN(C(=O)NCC(C)C)C2)=O)CCN(C(=O)Cc2ccns2)C1 c1(C(=O)NC(CN(C(C(CCSC)OC)=O)C)(C)C)ccc2nnn(O)c2c1 c1(OC)ccc(-c2ncccc2C(N2CC(C)NCC2C)=O)cc1[N+](=O)[O-] C1(C(N2CCCC3(CNC(C=CC)=O)C2C3)=O)CCC2(CC1)NC(=O)NC2=O C1(NC(CSCC#C)=O)CC(CCNC(C2(SC)CC2)=O)C1 C1(CC(=O)NCCN(C(=O)CCC2CC(F)(F)C2)CCOC)CCCC(F)(F)C1 CC(CC(=O)NC1CCC(NC(=O)CC(F)(F)F)C1)CC(C)(C)C C1(NC(CC=C=C)=O)CN(C(=O)CCOc2ccc(C(C)C)cc2)C2(CCC2)C1 C12(C(=O)NCC3(O)CC(C(=O)NCC(C(C)C)(C)F)C3)CCC(CC1F)C2 C(CCCCC(=O)N(C)Cc1ncccn1)N(C(C1C(C)CCCC1)=O)C C(=O)(C1OCCc2ccc(Br)cc21)N(C)CCNC(=O)C(C)(C)O N1(C(C(C)n2cncn2)=O)CCC(C2CCCN2C(c2cnn[nH]2)=O)C1 c1(OCCC)c(OC)cc(CNc2nc(OCC)cc(C)n2)cc1Br N1(C(Cc2cn(CC)nn2)=O)CC(CNC(=O)Cn2cnc(C(N)=O)n2)C2CC12 c1(CN(CC(C(=O)O)OC)C2CC2)ccc(Cl)cc1C CC(C)C(C)C(CNC(c1ccc(F)cn1)=O)NC(c1ccc(C2CC2)nc1)=O N1(C(C2C3CN(C(CN(C(COC)=O)C)=O)CC32)=O)CC(CO)CCC1C c1(NC(=O)NCC(C)N(c2ccccc2)C)ccc(-c2ccccc2)cc1F c1(C(=O)NC)cccc(C(N2CCCCC2C(C)NC(=O)CC(C)(C)SC)=O)n1 C(=O)(CCCCN=[N+]=[N-])NC1(CNC(C2CCC(CC)O2)=O)CC(OC)C1 C1(C)(C(N2CC(N(C)C(c3cccc(N4CCCC4=O)c3)=O)C2)=O)CCNC(=O)C1 S(=O)(=O)(c1cccnc1NCCc1nncs1)N(C(C)C)CCO c1(C(N2CCC(CN(C(C(CC)NC(C)=O)=O)C)C2)=O)cccc(Cl)c1 c1(CC)cccc(CC(=O)N(C)CCNC(=O)CC(C)C2CC2)c1 O=C1Cc2cnc(N3CCCC34CN(Cc3ccc([N+](=O)[O-])o3)C4)nc2N1 C1(C2CN(C(=O)CN(C(C3CC3)=O)CC)C2)(NC(CC(CC)OC)=O)CC1 C(=O)(C(F)C(C)C)N1CCC(C(C)(C)NC(C=CSC)=O)C1 Cc1ccccc1N(C)C(C1CN(C(=O)CC2CC(C)(C)CO2)CCO1)=O C1(NC(CCC)=O)(COC)CCN(C(=O)C(Cc2ccccc2)SC2CC2)CC1 C1(NC(=O)NC(c2cn(C)nn2)C)CCOCC1OC(=O)C(C)(C)C1CCCO1 c1(CC)nc(=N)[nH]c(=NCC2(CNC(C34CCCCC3OCC4)=O)CC2)[nH]1 CC1CN(C(=O)CSc2ccncc2)CCC1CNC(C1Cc2cscc2C1)=O N1(C(=O)Cc2nc(Cl)cs2)CCC2(CCCN(C(C3(O)CCC3)=O)C2)C1 c1(C(N2C(C)CCC(CNC(=O)CN=S(C)(C)=O)C2)=O)cc[nH]c2nccc1-2 C1(C(=O)NCCCC(=O)NC)CC2C=CC1N(C(C1(C)CC(OC)(OC)C1)=O)C2 n1(C(CC)C2CC2)nccc1C(N1CC(c2cn(CC3CCC(=O)O3)nn2)C1)=O C(C1=Cc2ccccc2OC1)=CC(=O)N(C1CCN(C(C2CNC(=O)C2)=O)CC1)C c1(C(N(C2CCN(C(=O)C(c3cncn3C)O)C2)CC)=O)ccc(CN(C)C)[nH]1 c1(OC)cncc(CC(=O)NC2CC(CO)N(C(c3nccnc3OC)=O)C2)c1 CC1CC(C(=O)NCC2(F)CC(NC(C3SCCS3)=O)C2)CC(C)(C)C1 CC(CO)CCN=c1[nH]c2c(c(=NCC3CC(C)(C)OC3(C)C)[nH]1)COC2 CC1CCCC(CC(=O)NC2CCN(C(c3snc(O)c3Cl)=O)C2)O1 c1(OC)ccnc(C(=O)NC2CC(CC(=O)NCCN(CC(F)F)C)C2(C)C)c1 c1(C(=O)NCC(C2CCN(C(C(CCC)C)=O)CC2)C)cc(C(F)F)cc(Cl)c1 C1(NC(CC2(C(=O)OC)CC2)=O)CC2CN(C(C3CC4CCC(C3)C4)=O)CC2C1 N1(C(c2c(OC)cc(CO)cc2)=O)CCC2CCCC12CC1(C(=O)NC)CC1 C1(NC(c2c(CC)noc2)=O)CC12CCN(C(=O)CCOCCOCCO)CC2 c1(OCC)cc(S(=O)(=O)N2CCN(C)CC2C)ccc1-c1cnc(COC)nc1 c1(C(=O)NCC(C2CC2)NC(C2C(C)(C)C2(F)F)=O)coc2c1C(=O)NCCC2 n1(CC=C)c(S)nc2cc(C(=O)NC(C(=O)O)C3CC3)ccc2c1=O C#CC1(C(=O)NCCc2cnn(C)c2C)CN(C(=O)CC(C)CN(C)C)C1 c1(C(=O)NC(CNC(c2c(C)nn(C)c2)=O)C(C)C)ccc2c(Br)cnn2c1 c1(C(C)C(=O)NC2CC2NC(c2ccn(CC#N)n2)=O)ccc(Cl)c(Cl)c1 N1(C(Cc2cn(C)nn2)=O)CC2CC(NC(c3c(F)ccc(F)c3Cl)=O)CC1C2 N1(C(C=C(COC)C)=O)CCCCC1CCN(C)C(C1(c2ccncc2)CC1)=O N1(C(C2(CN(C)C)CCC2)=O)CCCC1CNC(=O)CCc1cnoc1 CCC(CC(=O)N1CC(CNC(=O)CCc2cccc(O)n2)C1)C1CCC1 Cc1cc(C(N2CCOC(C)C2C(=O)NCCC(F)(F)F)=O)nnc1O c1(C(N(CCN(C(CCCOC)=O)C)C)=O)ccc(C)c(OC(F)F)c1.C(C)(=O)O CC1CC(F)(F)CCN1C(C1CC2CCC(C1)N2C(C1CNC(=O)N1)=O)=O N1(C(c2cc(C)cc(C)c2)=O)CC2(CCC(CNC(=O)CCNC(N)=O)O2)C1 O=[N+]([O-])c1ccc2c(c1)S(=O)(=O)CC2NCC1CC(F)(F)CO1 C1(NC(C2CC23CC(O)C3)=O)CCN(C(c2cnc(S)nc2)=O)CC1 N1(C(c2nc(CC)oc2C)=O)CCN(C(=O)CC23COC(CC)(C2)C3)CC12CC2 N1(C(CCC(=O)NCC)=O)CCC2(CC(NC(=O)CCC3(C)CC3)CO2)C1 Cc1cc(C(=O)NC2CCCC2CNC(C2C3CCCC23)=O)c2cnn(C)c2n1 Cc1nccnc1CCNCc1nnnn1C1CCC1.C1CCCCC1F C1(C(N(C)Cc2cc([N+](=O)[O-])ccc2Br)=O)CSC(c2cccs2)=N1 C1(COC)(NC(=O)C(CO)NC(N)=O)CCN(C(=O)C(C)OC(C)(C)C)CC1 N1(C(CC(c2ccccc2-c2nn[nH]n2)C)=O)CCC(C2CCNCC2)CC1 Cc1cnc(CCC(=O)NCC2CC(CNC(=O)C=CC3CCC3)CO2)[nH]1 Cc1cccc(CC(=O)NC2CN(C(=O)C(c3c(F)cccc3F)(F)F)C2)c1F N1(C(C2(CC)CCN(C(=O)COC3(C)CCC3)CC2)=O)CCN2CCCCC1C2 C1(C(=O)NC2(CNC(c3cncc(C4CC4)c3)=O)CC2)CCCS1(=O)=O CC1(C)CCN(C(=O)CC23CCCC2C3)C(C(N2CCCC3OCCC23)=O)C1 c1(C(C)(C)C)cc(C(=O)N(CCNC(C2CC(F)(CO)C2)=O)C2CC2)[nH]n1 CC1CN(C(C2CC(F)(F)C2)=O)CCC1N(C(=O)C(N)=O)C CCCN=C(NCCN1CCC(COCC)CC1)NC1CC(OC)C12CCCC2 c1(C(=O)NCc2cn(-c3ccc(OC)c(F)c3)nn2)cccc2c(Br)cccc12 c1(C(=O)NC(C2CCCCC2)c2nn[nH]n2)cc2c(Cl)c(Cl)ccc2[nH]1 C1(C(=O)NCC2(C)CCCNC2)CC(C2CCC2)C1 CCC(C)(C)C(O)C(=O)N1CC2CC2(NC(C2(c3ccc(OC)nc3)CC2)=O)C1 Cc1cc([N+](=O)[O-])ncc1C(=O)NCCCCNC(C1(C)C=CCC1)=O C12(CN(CC)Cc3ccco3)COCC1CN(C(C1CCCNC1=O)=O)C2 c1(NC(C2CCN(C(c3cc(Cl)n[nH]3)=O)CC2)=O)cnn2c1OCCC2 c1(C(CN(CC(N2CCOCC2)(C)C)C(C)=O)C(=O)N(C)C)ccncc1F c1(C(=O)NC2C(OC)CN(C(C3(Br)CCC3)=O)CC2)cc(F)cc([N+](=O)[O-])c1 C(C#Cc1cccc(OC(F)(F)F)c1)NCc1cn(CC)nn1 C(=O)(CC(C)CCCCCCCC)NCCCN(C(C(CC=CC)C)=O)C(C)C N1(C(C(CC(C)C)C)=O)CCC2(CC1)CCN(C(C13CC4CC1C3C4)=O)CC2C N1(C(COCC(=C)C)=O)CC(NC(=O)COCc2ccc(OC)nc2)C(C)(C)C1 c1(C(=O)NCC2(NC(C(N3CCC(C)C3)=O)=O)CCC2)cccc2nn(C)cc12 c1(C(N(CCC(C)NC(c2cccc(C)n2)=O)C)=O)c(N)cc(Cl)nc1Cl c1(OC)ccc(F)c(CN2CCN(C(C3(O)CC3)=O)C3CC23)c1 C1(CCC)(NC(=O)C=CCF)CCCN(C(=O)CCn2cccn2)C1 c1(NCc2c(C)scc2)cc(=NC2CCC(C)C2)[nH]c(C(C)C)n1 c1(CC)nc2sccc2c(=O)n1NC(=O)c1cnc(C(F)(F)F)cc1C Cc1c(C(=O)NCC2(C)CC(NC(c3coc(C#N)c3)=O)C2)cnc2ncnn12 Cc1c(C(F)(F)F)cc(Cl)c(Cl)c1NC(=O)Nc1cc(Br)ccc1I Cc1ncc(C(=O)NC2CN(C(=O)CNC(c3ccncc3)=O)CC2C)cc1N C(=O)(CS(=O)(=O)CCO)NC(C1CCOC1)CNC(c1cc(C)nn1C)=O C1(CNC(CC2C(C)CCO2)=O)CN(C(c2cnn(C)c2Cl)=O)CCN1C c1(CC(N2C(CN(C(CC)=O)CC)CCC2)=O)cncc(F)c1 N1(Cc2cn(C)nn2)CCN(C(c2cc(C3CC3)ncn2)=O)CC1 c1(C(=O)NCC2(CNC(c3ccn(C)c3)=O)CCC2)cc(Cl)c2ccccc2n1 S(=O)(=O)(c1ccc(C(C)(C)C)cc1)N1CCC(N(c2nccc(C3CC3)n2)C)C1 Cc1coc(C)c1C(=O)NCC1CCC(N(C(=O)C(C)CC2CCCC2)C)CC1 c1(OC(C2(C=C)CC2)=O)cccc(CNC(=O)CCCOCCOCC)c1 c1(OC)ccc(C(CNC(C2CCSC2)=O)NC(=O)Cc2cncn2C)cc1 N1(C(c2ccc(C(C)C)cc2)C)CCC(NC(c2cncn2C)=O)C(C)C1 CC(C)C(C(=O)N1CC2CCCC1(CNC(=O)C(C1CCOCC1)O)C2)C(C)C N1(C(CC(C)F)=O)CC(F)CC1CN(C(=O)CCCc1cccc(Br)c1)C C1(NC(C(CCC)F)=O)CCCN(C(c2cn(C3CC3)cn2)=O)C1CC c1(C(=O)NCC(C)N(C(C2CN(CCOC)C(=O)C2)=O)C)cccc2occc12 c1(CC(N2C(CNC(C=CC=CCC)=O)C(CC)CC2)=O)ccc(OC)cc1F c1(C(=O)NC2C(C)(C)CN(C(=O)CC3(O)CCC3)C2)c[nH]c2cc(C#N)ccc12 Cc1nc(N2CCCC(C(N3CCC(C)C3)=O)C2)c2ccccc2n1 C=CC1CCCN(C(=O)C(CC(C)C)NC(c2cc[nH]c2CCC)=O)C1 CC1(C)CC(C(N2CCOCC(NC(c3cnccc3C#N)=O)C2)=O)CCO1 C1(CNC(c2ccc(COC)o2)=O)CC2CC1CN2C(=O)CC1C(=O)NN=C1C S(=O)(=O)(c1ccc(Cl)cc1)NC1(C)CN(C(=O)CN2CCc3sccc3C2)C1 N1(C(C2CN(CC)C(=O)CC2)=O)CCC(NC(c2nonc2N)=O)C2(CCC2)C1 N1(C(C(C)Cn2cccn2)=O)CCC(C(=O)NCC2CCCCC2)C2OCCC12 Cc1cc(C(=O)NC(CC2CCC2)C(N2CC3CCC3(C)C2)=O)ccc1O C1(C(=O)NCCC(C)C(C)(C)C)C2CC(O)C(C2)N1C(=O)CC1(C#N)CC1 C(=O)(C1=C(Cl)CCC(C)C1)N1CCC2C(NC(COCCCC#C)=O)C21 N1(C(Cc2cc(OC)no2)=O)CC2(CNC(C3CC4C=CC3C4)=O)CCC1CC2 Cc1nccc(C(N2CCC(F)(CNC(c3ccc(F)s3)=O)C2)=O)n1 C(=O)(CCC(C)CN(C)C)NC(C1CCN(C(=O)C(C)(C)C#N)CC1)C C(CC1CCC1)(C(=O)NCCC1CC(O)C1)NC(C1C(=C)C1)=O C(CCC(C)(C)NC(=O)C(C)Cc1ccccc1Cl)NC(c1scc(C)c1)=O C(=O)(C1=Cc2cc(Cl)ccc2OC1)N1CC(C(C)NC(CCC#CC)=O)OCC1 CCC(C)C(=O)C(=O)N1CC2CC2C1C(N1CCC(C)(O)C1)=O c1(C(=O)NCC(CC(C)C)NC(=O)C(C)OC(C)(C)C)cnc2cc[nH]c2c1 N1(C(CCSC)=O)CC(CCNC(C2(c3ccccc3)CC2(F)F)=O)C(C)C1 C(CC(=O)NCC1CC(=C2CCC2)C1)(C(F)(F)F)NC(C=C(CC)CC)=O C(=O)(C1=Cc2ccccc2C1O)NCCC1(O)CN(C(C(CC)(C)F)=O)C1 C(=O)(C(C)(CNC(=O)CC(=O)NCC)CC)NC(CC=C)C1CC1 n1(C(C)C)ncc(Cl)c1C(=O)N(C(C)CNC(=O)CCCCc1cnc[nH]1)C c12cccc(c1)C(=O)N2.C(C(C)(C)C)OCC(=O)NC1C(CCOC)C1 c1(OCC)cc(CN2CCOC(CNC(=O)CCCCCl)C2)ccc1OC C(c1ccco1)=CC(=O)NCCCOCCC(=O)NC(COC)CO CC1CCC(C)(C(=O)N(CCNC(=O)CCOCC(F)F)C2CC2)C1 N1(C(C2(C#N)CCCC2)=O)CC2CC(NC(C3CCC3(F)F)=O)C1C2 C1(CNC(C(CC)(C)CO)=O)CN(C(c2scnc2C(F)F)=O)CCC1(C)C c1(C(N(CC(CN(C(c2cnc(C)s2)=O)C)O)C)=O)cc(N)cc([N+](=O)[O-])c1 C(=O)(CCC(C(C)C)NC(c1c(C)n[nH]c1C)=O)NCC(=O)OCC=C c1(C(=O)NCC2(F)CC(NC(C3CCCCC3O)=O)C2)cncc2c1CCCC2 c1(C(=O)NCCOCCN(C(=O)CN2CCCCC2)C)cccc2c1OCCC2 N1(C(c2c(CC)csc2)=O)CCCN(C(C2CCOC(C)(C)C2)=O)C(CO)C1 c1(C(=O)NCC2(C(=O)NOCCC3CC3)CCCO2)cc2ccncc2[nH]1 c1(C(N2CCN(CC)CC2)=O)cnc2[nH]cc(-c3cc(F)ncc3OCC)c2c1 C(C(C(=O)NC(CSC)C(F)F)n1cc(CCc2ccccc2)nn1)OCC c1(C(=O)NC2CN(C(c3nn[nH]c3Cl)=O)C2)cnc(C2CC2)o1 N1(C(c2[nH]cc(C)c2)=O)CC(C(=O)NCC2(C)CC3CCC2C3)CC1(C)C CC(C)(CC(=O)N1CCC2C(NC(=O)C=CC3CCCCC3)C2CC1)CC(F)F C12(NCC3CC3)CN(C(CC3CCCN(C(=O)OC(C)(C)C)C3)=O)CC(F)(C1)C2 c1(C(N(C2CN(C(c3nc(C)[nH]n3)=O)C2)C)=O)ccc(CNS(C)(=O)=O)cc1 N1(C(Cc2nc(CC)sc2)=O)CCCCC1C1(NC(=O)COC(C)=O)CC1 CC(C)S(=O)(=O)C(C)C(=O)NCCN1CCN(C(=O)COC2CC2(F)F)CC1 C1(C2CCCN(C(c3n[nH]c(=N)s3)=O)C2)(NC(CNC(CC)=O)=O)CC1 C(=O)(C1CCCc2sccc21)N(CCOCCCNC(C(CC=C)C)=O)C c1(C(=O)NCCC2CC(NC(c3cc(C)oc3C)=O)C2)nc(C)n(C2CC2)c1C Cc1cccc2nc(N3CCOCC(NC(c4coc(Cl)c4)=O)C3)oc12 C1(C(=O)OC)(C(=O)NC2CC2CNC(C2CC(F)(F)C2)=O)CCCC1 c1(OC)nc(C(C)C)ccc1-c1ccc(C(N2CCC(C(N)=O)CC2)=O)nn1 c1(C(N2CCC(O)(CCNC(C(CC)OCC)=O)C2)=O)cnc(C)c(N)c1 c1(C(N2CCC(C)(NC(CC3(C=C)CC3)=O)C2)=O)ccc2cccc(O)c2c1 CC12CC(C(N3CC(F)(F)CC3CNC(c3coc(CO)c3)=O)=O)(C1)C1(CO1)O2 c1(-c2onc(Cc3c(C(C)O)ncc(Br)n3)n2)cnc2c(F)c(F)ccc2c1 C(CCCCCN=c1cc(C)nc(N2CCn3ncc(Cl)c3C2)[nH]1)SC Cc1nn(C(C)(C)C)cc1C(N1CC(NC(=O)C(C)(C)CN(C)C)C(F)C1)=O CCCCCCC(CC)C(=O)NC(CO)CCCCNC(=O)C=C(C)Cl CC1=C(C(=O)N2CCN(C(=O)C(N3CCCC(C)C3)=O)CC2COC)CCCO1 c1(C(=O)NCCN(C)C(C2CCC(c3ccccc3)CC2)=O)cc(N)cc(O)n1 c1(N2C(CNC(CC3(OCC)CCC3)=O)CC3(CC3)C2)nc(C)nc(Cl)c1CC C1(C(N2CCCC2CN(C)C(C23CC(CN2C2CC2)C3)=O)=O)(CC)CC(C)(C)C1 N1(C(C2CCCN(CC)C2)=O)CC2OCCN(C(C3(c4ncco4)CC3)=O)C2C1 C1(NC(C(C(C)C)N(C)C)=O)CCCN(C(=O)CC2COCCOC2)C1C c1(CC(C(=O)NCC(c2ccc(C)cn2)OC)(C)O)ccc(O)c(O)c1 c1(C(N(CC(C)NC(C2(CSC)CC2)=O)C)=O)ccc(Cl)c(C)c1 C1(NC(c2ccc(CNC(CN3CCC(=O)CC3)=O)nc2)=O)(CO)CC2CCCC12 Cc1c(C(=O)NCCCN(C(c2ccnc(S)c2)=O)C2CC2)cnn1C(C)C C1(NC(=O)C=CCO)CN(C(C2CCCN2CC2CCCC2)=O)CC2(CCC2)C1 C1(NC(Cc2ccn(C)n2)=O)CCCC12CN(C(=O)CCC1CCCO1)C2 N#Cc1ccc(CC(N2CCCC(CNC(C3CCC(CO)CC3)=O)C2)=O)cn1 c1(C(N2CCC(N(CCC)C(c3cnc(O)o3)=O)C2)=O)cncc(Cl)c1 O=C(C(CNC(C1(O)CC1)=O)Cc1ccccc1)NCC1=CCCCC1 CCC(CN(C)C)C(=O)NC1CCCCC1CNC(=O)C(=O)NCC(F)F c1(OC)ccc(-n2nc(CC(C)(C)CO)nc2CCC2CCCCC2)cc1 c1(CC(=O)NCC(C)CNC(C2CCC2)=O)csc(NC=O)n1.c12ccnn1C2 C(C(C)N=c1[nH]ccn2nnnc12)N(C(CC=C)=O)C Cc1cc(C(=O)NCC(C)CN(C(=O)CCc2cc(C)on2)C)cc(Br)c1 c1(C(N2CCN(C(COCCC=C)=O)CC2COC)=O)cccn2cc(C)nc12 C(=O)(CCN=C(NCCC(F)F)NCC1CCCC(C)(C)C1)N(C)C C1(NC(C(C)N(CC)CC)=O)CC2CCC1CN2C(=O)Cc1cnns1 C=CC1(NC(N2CCC(C(=O)O)C(C)C2)=O)CCCCC1.c12ccccc1S2 C(=O)(C(C#N)C1CC1)NC(C)CN(C(=O)COCC1CCCC1)C C(=O)(CC(C(F)(F)F)NC(=O)C=CC1CCCN1C)N(C(C#C)C1CCC1)C NS(=O)(=O)CC(=O)NCC(c1ccccc1)NC(=O)CCc1cccnc1 c1(C(=O)NC2C3(CC(NC(Cc4cccc(C)c4)=O)C3)C2)c(O)nnc(C)c1C c1(OCC)ccc(Cl)cc1C(N1CC2(C1)CN(C(c1ccc(O)c(C)c1)=O)C2)=O CCS(=O)(=O)CC(=O)NC1CC=C(C(=O)NCc2ccc(F)cc2F)C1 Cc1nc(O)[nH]c1C(=O)NC(C1CCCCN1C(=O)CCc1cc(C)n(C)n1)C Cc1cc(C)n(-c2ccnc(NC(=O)CCC(C)NC3(N(C)C)COC3)n2)n1 c1(NC2(CNC(c3scc(OC)c3)=O)COC2)ncc(Cl)cc1[N+](=O)[O-] CC(C)C(C)C(C)CC(=O)NC1(CO)CCN(C(c2ccn(O)c(=O)c2)=O)CC1 CC(C)C(C)C(CNC(=O)CN1CCN(C)CC1)NC(=O)CCF Cc1ccc2c(c1)CC(C(=O)NC1(C)CCCN(C(c3[nH]c(C)nc3C)=O)C1)S2 N1(C(CC(C)C2CC2)=O)CCC2(CCCN2C(C2CCC(N(C)C)CC2)=O)CC1 C(CC#CC)(C(=O)N1CC(c2ncc[nH]2)C1)NC(C1CCC(=C)CC1)=O N1(C(c2c(C)nc(CCC)s2)=O)CCCC(C)C1CNC(=O)C=CC(F)(F)F C1(NC(=O)C(=O)N(CCCNCC)CCO)Cc2cccc(OC)c2O1 [N-]=[N+]=NC1COCC1NC(=O)C(Cn1ccnn1)NC(=O)CCn1cnc(=N)[nH]1 c1(CC(N2CCC(N(C)Cc3c(OC)nccc3)C2)=O)cc(Br)ccc1Br CC(F)(F)C(F)C(=O)N(CCCNC(C1(C)CCNC1=O)=O)CCO C1(NC(C(C)N(CC(F)(F)F)C)=O)CCCC(CNC(=O)CC2CC3(CC3)C2)C1 C1(C(=O)NC2CCC(NC(c3ccc(NC(C)=O)cn3)=O)C2)CCCCS1(=O)=O c1(NC(=O)CCC(=O)N2CC(Oc3nccs3)C2)c(Br)cc(F)c(F)c1F CC(c1ccccc1)=CC(=O)NC(C)CN(C)C(c1cnc(N(C)C)nc1)=O N1(C(c2cn(CC)nc2)=O)CC(C)OC2(CCN(C(=O)CC(=O)N(C)C)CC2)C1 c1(NC(C(CC2CCOCC2)NC(c2ccc(O)nn2)=O)=O)ccc(F)cc1O Cc1ccc2c(c1)c(=O)n(C(C)C(N)=O)c(=O)n2C.C123CC(C1)(C(C)O2)NC3 C(=O)(C1CCCc2nn(C)cc21)N1CC2CCN(C(C(CC)CC)=O)C2C1 C1(CNC(c2c(C)ccc(C)c2)=O)CN(C(c2nscc2C)=O)CC(C)(C)C1 C1(C(N2CC(C(C)NC(c3nncn3C3CC3)=O)C2)=O)CCc2nncn2C1 C(=O)(CC(C1CC1)NC(=O)C(C)NC(C)=O)N(C(CC)CC)C O=C(CCC(=O)c1cccc(F)c1)NC1CC(CNC(C23CCC(C2)C3)=O)C1 N1(C(C2CC(OC)C2)=O)CCOCC1.N1(CC)CCNC1=O CC1(C(=O)NCCCCC2CCC2)CC(O)CN1C(C1CC1(C)C(F)F)=O Cc1c(C(N2CCC2Cn2cc(C3CCCOC3)nn2)=O)sc2cncn12 CC1=NS(=O)(=O)NC(C)=C1CCC(=O)NC1CC(NC(C2(Cl)CC23CCC3)=O)C1 n1(CC(N2C(C(C)NC(c3c(OC)csc3)=O)CCC2)=O)cnccc1=O CCCC(C)(C)C(=O)N1CCC(C)C1C1CCN(C(=O)CCC(C)(C)OC)CC1 C=CCC(CC=C)C(=O)NCC(CCC)NC(=O)CCC C12(C(=O)NC3CC(F)(CNC(c4cnc(O)c(F)c4)=O)C3)CCCC1C2(F)F C1(C(=O)NOCCCO)(CC=C)CC=CC1.C12CCC(C1)C(=O)N2C1CC1 CC1=NOC(C)(C(N2CC(CNC(C3(C(F)F)CCOCC3)=O)C(O)C2)=O)C1 C1(CNC(c2c(C(C)C)nns2)=O)(CNC(=O)CC2CCOC2=O)CCCCC1 N1(C(C=Cc2c(C)ccnc2)=O)CCCC12CCN(C(C1(F)CCOC1)=O)CC2 c1(OC)ccc(=NC(=O)C2CC2NC(=O)C=Cc2ccc(Br)cc2)[nH]n1 CCCCC(C(=O)N(CC(N1CC(C)OCC1C)=O)CC1CC1)C(C)C c1(C(=O)NC(CC)(C)CNC(c2ccc(C3CC3)cn2)=O)cc(O)nc(OC)n1 c1(CC(=O)NC(CC2CN(C(C3(OC)CC3)=O)C2)C)csc2ccc(C)cc12 CCCCC(C)C(=O)NCCN(CCCCCC)C(C1CN(S(N)(=O)=O)C1)=O C1(C(=O)NCC(CNC(c2c(COC)cc[nH]2)=O)(C)F)CC2CC(=O)C1C2 c1(C(=O)NCC23C(CN(C(c4cnc(C(C)O)s4)=O)C2)C3)cnc2[nH]cncc1-2 c1(OC)cc(C(N2CC(O)C(O)C2)=O)cnc1-c1ccc(OC2CC2)cc1 C1(CNC(Cc2cncc(C)c2)=O)CN(C(c2cncc(N)c2)=O)CCN1C C(=O)(CCCN=[N+]=[N-])NCC1CCN(C(CCn2c(C)ncc2)=O)C1 c1(C(N(C)C)=O)nn(C)cc1C(=O)NCCN(C(=O)C(C)(F)F)C C1C(=O)CCN=C2N=c3sccc3=C(N2)N2CCCC(C2)CN1.N1(CC)CCC1 c1(C(=O)NC2CN(C(COC)=O)CC2CC2CC2)nn2cccnc2c1Cl CCC(CC)(CO)C(=O)N1CCC(O)(C(C)NC(=O)CCNC(C)=O)C1 CCC(C)(CO)C(=O)N1CCCC(NC(=O)CCc2cn(C)cn2)CC1 c1(OC)cc(CC(=O)NC(CO)C(C)NC(C2CCC2)=O)ccc1C c1(OCCC)cccc(CC(=O)NC2CCC2NC(=O)Cc2cc[nH]c(=N)c2)c1 CC1(C)C2CCC(C(N3CC(F)CC3CNC(C3CCCO3)=O)=O)C1C2 N1(C(Cc2ncc(CC(=O)OC)[nH]2)=O)CCC2CN(C(=O)CCC3(C)N=N3)CC12 CC1(C)CC(C(=O)NC2(C3CN(C(=O)CC4C=CCC4)C3)CC2)CC(C)(C)O1 C=C(C)CCCC(=O)NCC1COCCN(C(C2CC(S(C)(=O)=O)C2)=O)C1 c1(OC)ccc(F)c(C(=O)NCC2(NC(=O)COCP(C)(C)=O)CCCC2)c1 c1(C(CC)C)cccc(C(=O)NCCC2CC=CC2)c1 C(CCN=c1cc(C)c(S(=O)(=O)NCc2cn(C)nc2Br)c[nH]1)SCC=C CCC(O)C(F)(F)C(=O)N1CC(c2cnnn2C)(N(C)C)C1 c1(C(N2C(C)CCC2C(=O)NC(c2ccccc2)C#N)=O)cc(F)cc(Br)c1Cl c1(C(N2CCCC2Cc2ccc(C)cc2)C(=O)NC)cccc2[nH]ncc12 Cc1cc(O)c(C(=O)N(CCCCNC(=O)CCP(C)(C)=O)C)cc1Br C1(NC(Cc2nc(CC)sc2)=O)CCS(=O)(=O)C12CN(c1ncccc1C#N)C2 c1(C(=O)NC(CCNC(C(C(CC)C)OC)=O)(C)C)coc2c(OC)cccc12 C1(N(C(CC(C)C)=O)C)CN(C(=O)C(C)COc2ccccc2)CC1(C)C CC1CC(C(=O)N(C)CC2CN(C(=O)CCC3CCCO3)C2)CC(C)(C)C1 N1(C(C2C(c3ccc(OC)cc3)C2)=O)CCN(C(=O)C(C)S(C)(=O)=O)C(C)C1 CC1CC(NC(c2snnc2C2CC2)=O)CN(C(=O)CCn2cncn2)C1 S(=O)(=O)(c1ccc(OC)nc1)N1CC(CC(=O)OC)OC(C)(C)C1 CCCCC(C(=O)NCCCC1(NC(c2cocc2C)=O)CC1)C(C)C C(C)(C(C)(C)NC(=O)CSC(F)F)NC(CCN(CCC)C)=O C(=O)(C(C)(C)C(C)(C)O)NCC1N(C(C(C(C)C)c2cnc(C)s2)=O)CCC1 N1(C(CNC(CC)=O)=O)CCCC(N(C(=O)C2=CCCCC2)C)CC1 c1(C(=O)NCCNC(C=Cc2n(C)cnc2)=O)ccc2nc(C(F)(F)F)[nH]c2c1 CC1=C(C(=O)NCC2(F)CN(C(C3C4CC5C(C4=O)C35)=O)C2)CCC1 c1(C(=O)NC2CC2(F)F)c(NCc2cccc(Cl)n2)sc2c1CCCC2 N1(C(c2c(C)occ2)=O)CC(CNC(=O)CCOc2cccc(F)c2)C(C)(C)C1 NS(=O)(=O)CCCCCC(=O)NCCCCNC(c1ccnc(Cl)c1F)=O N1(C(Cc2n(C)cnn2)=O)CC2(CC(NC(C3(C)CCC(=O)NC3)=O)C2)C1 c1(CNC(C(=O)Nc2c(C(=O)OC)c(-c3cccs3)cs2)=O)nc2c(o1)CCSC2 C1(C(N2C(C)CN(C(=O)C3=C(Cl)CCCC3)CCC2)=O)CSC2(C)CCC(=O)N12 c1(C(C)=O)cc(C(=O)NC2CCCC2NC(=O)CNC(=O)C2CC2)c(C)o1 N1(C(c2cnn(C)c2Cl)=O)CCCC2CN(CCc3cc(Cl)cc(Cl)c3)CCC12 C1(NC(C(C)SC)=O)C2CC3C(C2)C13C(=O)N(C)CC1CCCC1(C)C CCC(CC(F)F)C(=O)NCC(C)(C)CN(C)C(c1cc(C(F)(F)F)ns1)=O N1(C(C(CC)(C)C#N)=O)CCC2(CC1)CC(C)N(C(c1ccc(F)c(Cl)c1)=O)C2 N1(C(c2ccc(Cl)s2)C(=O)NC(CC)C)CCOCC1CC(=O)OC C(=O)(CCCCC#N)NCC(C)NC(C(=O)NC)=O N1(C(Cc2ccn(C(C)C)n2)=O)CC2CC(NC(=O)COCCOCCO)C1C2 c1(C(=O)NCC2CN(C(c3ccc(OC(CC)C)cc3)=O)C2)cc2scnc2[nH]1 C(CC(C)(C)C(=O)N1CCC(O)C(F)C1)NC(CCNC(=O)NC)=O Cc1nc(C(=O)NCCC(C)NC(=O)C(O)CC(F)F)c(C)n1C1CC1 c1(C(N2CC(c3cn(CC(CC)C)nn3)C2)=O)ccc2[nH]ccc2c1F N1(C(C=COCC)=O)CC2CCCCC2(CNC(=O)C2=CCOC2)C1 CC#CCCCCNC(c1cccc(C(=O)NC2(c3ccccc3)CC2)n1)=O N1(C(CCCCC(=O)NCCC)=O)CCC2(CCCC2NC(c2ccoc2)=O)C1 CCCCC(=O)C(=O)NC(C(=O)NC(c1cc[nH]n1)C)c1ccoc1 C1(NC(=O)CCc2cccnc2)C2CC(CN(C(=O)CCC3CCC3)C2)C1CO C1(NC(c2c(C)c[nH]c2)=O)CCCC(C(N2CC(CC(C)(C)C)C2)=O)CC1 C1(F)(C(=O)NCCCC2N(C(=O)OC(C)(C)C)CCC2)C2CCCC12 C(=O)(C(CC)C(=O)NC1C=CCCC1C(N1CCCC(C(=O)OC)C1)=O)OCC C(=O)(C1=CCCC1P(C)(C)=O)N(C(CNC(c1c(SCC)nccn1)=O)C)C C12(NC(N)=O)OC3CC4CC(C5C4C3C15)C2.C1(=O)CN1C(C)C.C(=O)(C)NCC C1(CNC(C2C(OC)C2)=O)CN(C(=O)CCn2cnnn2)CC2(CCC2)O1 C1(CNC(CC(CC)C2CCC2)=O)CC2(CCC2)CN1C(=O)C=CBr CC1OCCN(C(c2cc(C#N)cn2C)=O)C1C(=O)NCCC(C)(C)N(C)C C1(NC(c2[nH]cc(C)c2)=O)CN(C(c2coc(Br)c2)=O)CCC1F C(=O)(CCCC(C)(C)C)N1CC(N(C(=O)C(c2cccc(Cl)c2)O)C)C1 n1(CCC(=O)Nc2cncc(C(N)=O)c2)ccc2cccnc12 N1(C(c2c(C)cccn2)=O)CC(C)CCC1CNC(=O)CCc1nnc(S)n1C C(=O)(C1=NOCC1)NCC(CNC(Cn1c(CCC)ncc1)=O)O C1(C(=O)OC)CC2CC1CC2.N1(C=O)CC2C(C(=O)N(C)C)C2C1 CCCCC(CC)CC(=O)NCCC(C)(C)C(=O)NCc1coc(C)c1 c1(C(N(CC(C)NC(=O)CN2CCSCC2)C)=O)ccc(=O)n(CCF)n1 C12(CNC(C3CCC4(CC3)CC4)=O)CN(C(=O)CC3=CCCC3)CC1CCO2 c1(CN(C(=O)CN(C)C)C(C)C)nncn1C n1(CCC(=O)NCCC2N(C(COC)=O)CCOC2)cnc2c(cnn2C)c1=O C1(NC(C23N(C(COCC(=C)C)=O)CC(C)(C2)C3)=O)CCc2nn[nH]c2C1 Cc1c(C(N2CC(NC(c3nnc(C(C)(C)C)s3)=O)C2)=O)nnn1C Cc1cc(Cl)c(C)c(C(=O)N(C)CC2CCN(C(=O)CCc3cscn3)C2)c1N C1(NC(c2cccc(NC(Cn3c(C)ncc3)=O)c2)=O)(CO)CCC(C)(C)C1 CS(=O)C1CN(S(=O)(=O)CCCC2CC2C)C1 Cc1cc(C)nc(NNC(=O)NC2CC(CC#N)C2)c1 Cc1ccc(C(N2CCCC(O)(CNC(=O)CC3CCCCO3)C2)=O)cc1O c1(CN2CC(NC(c3cc(Cl)cnc3Cl)=O)C(O)C2)ccn2ccnc2c1 c1(C(=O)NCC(CNC(CC2CC(=C)C2)=O)C)nc(O)nc(O)c1F C(CC(C(C)(C)C)NC(c1cn2ccsc2n1)=O)N(C)C(c1csc(O)n1)=O C(C(C)C)(C(O)C(=O)NCC1CCN(C(=O)C(C)OCC(C)C)C12CC2)OC c1(C(=O)NC(C2CN(C(C3(C=C)CCC3)=O)C2)C)csc2cc(Cl)cnc12 c1(C(=O)NC2CCC(CCNC(=O)CNC(C3CCCC3)=O)C2)cccc(F)c1 C1(CC)CCCC1(C)C(=O)NCCN(C(=O)CCNc1cccnc1)CCOC CCC(CC)(CO)C(=O)N1CCCC(O)(CCNC(=O)C2=NNC(=O)CC2)C1 N1(C(C23CC(C)(C2)C3)=O)CCCC1C1CCCN1C(=O)CCCN1CCCC1 c1(C(CNC(c2csnn2)=O)NC(c2cn(CC=C)nn2)=O)ccc(F)cc1F c1(C(=O)NC2C(NC(C3CNC(=O)N3)=O)CC2)ccc(F)c(O)c1F N1(C(C(c2c(C)nn(C)c2)=O)=O)CCC(NC(=O)CN2CCN(C)CC2)C1(C)C C1(NC(Cc2cccc(CC)c2)=O)CCN(C(C2CCCC(F)(F)C2)=O)C12CC2 C(=O)(C(C#N)C(C)(C)C)NC(COC)CC(=O)NCc1cccnc1Cl c1(C(=O)NCC2(C)CCC(NC(C(C)(C)Cc3cnn[nH]3)=O)C2)cc(Cl)nnc1O c1(C(=O)NCCC2OCCN(C(C3C(C)(C)CO3)=O)C2)ccc([N+](=O)[O-])[nH]1 N1(C(C(CC)(C)OC)=O)CC2CC(NC(c3cc(C(C)C)nn3C)=O)CC2C1 S(=O)(=O)(c1cccc(Cl)c1)N1CC2CN(Cc3ccc(OC)nn3)CC21 C12(C(N(C3CCCN(C(=O)C=Cc4cscn4)C3)CC)=O)CCCC1C2(F)F c1(SC)ccc(C(N2CCC(C(F)C(=O)NCCC3CCN(C)C3)C2)=O)o1 C(=O)(CCC(=O)NCCC1(NC(=O)CN(C2CCS(=O)(=O)C2)C)CC1)NCC C(=O)(C(C)Cn1ccc(C)n1)N(C(C)CNC(=O)C(n1cc(C)cn1)C)CC N1(C(CCCC=C)=O)CCN(C(=O)C2=CCCOC2)CC1CCCC c1(C(=O)NCCC(C)NC(CCc2c(C)cccn2)=O)ncc(Br)cc1N c1(NC(C(C)C)CNC(=O)Cc2ccc(O)nc2)nc2ncc(Cl)cc2s1 C1(NC(=O)OC)C2CC3C(C2)C13C(=O)NC(CNC(=O)Cc1csc(NC)n1)C N1(c2nc(C)nc(O)c2)CCCC(C2(NC(c3cc(C(F)(F)F)on3)=O)CC2)C1 Cc1c(C(N2CC(C)(C)CC2CNC(=O)C=CC(C)(C)C)=O)cccc1Cl CC1CC(NC(=O)C(=O)Nc2ccccc2O)CN1C(C1CC(O)C1)=O C(=O)(CCC1=NNC(=O)CC1)NCC1(CNC(c2ccc(CC)c(Cl)c2)=O)CC1 O=C1CCN(CC(N2CCC(C(O)CNC(c3cnsc3)=O)CC2)=O)CC1 N1(C(C(CC)O)=O)CCN(C(CNC(c2ocnc2C2CC2)=O)C(F)(F)F)CC1 C(=O)(C(CNC(c1coc(C(C)C)n1)=O)C(C)C)NCc1c(CC)cncc1 C1(CNC(CCn2c(C)ncc2)=O)COCCN(C(C2CC(C3CC3)=NO2)=O)C1 c1(CC)ccc(OCCC(=O)NC(C)(CNC(=O)C(F)(F)OC2CC2)CO)cc1 c1(N2CC(NC(C=COCC)=O)C(O)C2)ncnn2cc(Br)cc12 C1(CNC(C(C)SC(F)(F)F)=O)CCC(N(C(=O)C(C)OCC(F)(F)F)C)CC1 c1(N(CC(CNC(C2(CC)CC2)=O)C)C)nc(C)nc2scc(C)c12 C1(NC(CC2N(C(Cc3ncn(C)c3)=O)C3CCC2C3)=O)CC12CCOCC2 c1(C(N2C(CNC(CSC)=O)CCC(C)C2)=O)ccc(S(=O)(=O)NCCO)s1 C(=O)(C#CC(C)(C)C)NC1C(NC(C(c2scc(C)n2)C)=O)CC1 C1(CNC(c2c(C)nn[nH]2)=O)CN(C(=O)C(C)c2cncs2)C2CCCC2O1 N1(C(C(C)NC(=O)CC(F)(F)F)=O)CCCCC(CNC(=O)CC2CC=CC2)C1 c1(CC(N2CC(CC(C)NC(c3cc(O)ncc3F)=O)C2)=O)ccc(F)c(F)c1 Cc1cc(C)c(C(=O)NCCN(C)C(C2(C)CCCCC2(F)F)=O)c(S)n1 c1(CCC)ccc(C(N2CC(NC(c3cnnn3C3CC3)=O)C2)=O)s1 C1(NC(C(Cc2ncn(C)c2)O)=O)CCN(C(=O)C(=O)Nc2ncc[nH]2)C12CC2 C(=O)(CCC1=CCCCC1)N1C(CC)CN(C(=O)CCNC(N)=O)CC1 C1(C)(CC)CCCC1NC(=O)CC1CC1CNC(=O)CS(=O)(=O)NC N1(C(COCC)=O)Cc2nccn2CC(NC(=O)CCC(C)CC)C1 C1(NC(CN(C(C(C)C)=O)C)=O)CC(C)(NC(=O)COCC2CCC2)C1 N1(C(c2ccc(C)cc2C)=O)CCC(C2CCCN(C(C3CCCC3F)=O)C2)C1 N1(CC2CN(Cc3ccccc3)CC3(C2)CC3)CC2CCC1C(O)C2O c1(C(N2CCN(C(CC)=O)C(C)C2C)=O)c[nH]c2cc([N+](=O)[O-])ccc2c1=O N1(C(C2C(C#C)C2(C)C)=O)CCn2ncc(CNC(C3(O)CC3)=O)c2C1 C(=O)(C(F)(CNC(c1cc(C)co1)=O)C(C)C)N1CCC(CN(C)CC)C1 C12(C(C)=O)CCC(C(N3CCOC(CNC(C4CCCO4)=O)C3)=O)(CC1)CC2 Cc1cc(C(=O)NC2(C(=O)NCCC3CCCN3C)CC2C)no1 C=CCN=C(NCC1CC(=O)c2ccccc2O1)N1CCN2C(=O)NCC2C1 C1(C(F)(F)F)(C(=O)NCc2cn(-c3ccc(F)cc3Br)nn2)OC2CCC1CC2 c1(CNC(C(C2(C)CC2)NC(C(COC)OC)=O)=O)cncc(F)c1 c1(C(=O)NCC2OCCN(c3snc(COC)n3)C2)coc2c1CCCC2 C(N=c1nc(CC2CC2)[nH]s1)C1C(NC(C(C(C)C)n2cnnc2)=O)CCCC1 C=CCC(CNC(c1c[nH]cc1CC)=O)C(=O)NC(C)(CO)CCCC C(=O)(CCCCCC(C)C)NC1CC2(C(C(N3CC(OC)C3)=O)C2)C1 N1(C(c2ccc(N(C)C)cn2)=O)CCC2CN(C(C3CN(S(N)(=O)=O)C3)=O)C2C1 C1(SC)CN(C(=O)CC2(C)CC2(Cl)Cl)CC1NC(C1(n2cccn2)CCC1)=O C(=O)(C#CC(C)(C)C)N1CCCC(N(C(C(C(C)C)C)=O)C)C1 C1(CC(C)NC(=O)C(=O)NC2CC2)CC2CCC(C1)N2C(c1cc(O)cc(O)n1)=O N1(CCCNCC2CCN(C(=O)OC(C)(C)C)C2)CCC(S)c2ccsc21 c1(CC)ncc(C(N2CC(F)CC2CNC(C2C3COCC23)=O)=O)c(O)n1 C1(CNC(CC=CC=C)=O)COCCN(C(=O)C(C(C)(C)C)NC(C)=O)C1 N1(C(CC(C(C)C)(F)F)=O)C2CCC1CN(C(c1ccsn1)=O)CC2 C1(c2c(C)ncs2)CCN(c2ccnc(NC(c3ncccc3F)C)n2)CC1 N1(C(C2(C)CC2Br)=O)CCCC2(C1)CN(C(=O)CCc1nc(O)n[nH]1)C2 Cc1cc(Cl)cc(NC(C2CC2C(=O)Nc2ccc(Br)s2)=O)c1I C(=O)(C1CCCn2ncnc21)NCCCCC(C)NC(C1CCC(C)CC1)=O c1(OC)ccc(C(O)C(=O)NC2CCCC2CNC(C2(CO)CCCO2)=O)cc1 C1(NC(C2CC=CC2)=O)CCCCC12CCN(C(C1CC13CC(F)(F)C3)=O)CC2 C1(C2CCC2)(C(N2C(CNC(c3ccc(F)cc3)=O)CC2)=O)CCC1 C1(C)(CNC(CN(C(C)C)C)=O)CN(C(=O)Cc2cn(C)cn2)C(C)(C)C1 N1(C(c2ccncc2Br)=O)CC2CN(C(C3CC3(F)F)=O)CC2C1 Cc1ccc(C(=O)NCC23CC2CN(C(=O)CCN2CCCCCC2)C3)nc1O N1(C(C(c2nccc(C)c2)(C)C)=O)CCCCC2(C1)CN(C(C1(C)CC1F)=O)C2 CC(C)CC(C(=O)NCC1CCOCC1)ONC(C1(O)CCSC1)=O n1(CC)nc(C)c(C(=O)NCCCCCN(C)C(C2CCCOCC2)=O)c1Cl C(=O)(C(C)CCC(C)(C)C)N1C(CC)CN(C(C2CCC(CCO)CC2)=O)CC1 N1(CCC(=O)NC(CN(C(=O)CCc2ccccc2)CC)C)CCCCC1=O C1(CNC(COCCCC)=O)CN(C(=O)CCc2ccc(C(=O)O)[nH]2)CCCO1 CN=c1[nH]nc(CC(=O)NCCN(C)C(C2COC(C)C2)=O)s1 N1(C(c2n(OC)cnc2C)=O)CCC2(CC1)CC2CNC(C1(Br)CC1)=O C#Cc1ccc(OC)c(C(=O)NCC(C)CN(C(=O)CC2CC(=O)NC2=O)C)c1 N1(C(c2c(CC)cccc2F)=O)CC2OCCN(C(=O)CC(C)CC)C2C1 C1(COC(CCC=C=C)=O)CCC(=O)N(C(=O)C=C2CCCCC2)CC1 C1(C(N(CC(CN(C)C(c2c[nH]nc2C2CCCO2)=O)O)C)=O)CC=CCC1 Cc1cnc(CNC(=O)NC(C2CCC2)C2CCC2)c(C)c1 C1(CC(=O)N(C2(CNC(C3CCCCS3)=O)CCC2)C2CC2)CC2CC2C1 CC(C)(CCNC(=O)COC1CCOC1)NC(C1CN(C2CCC2)C1)=O c1(C(C(=O)NCC(C)CN(C)C(c2coc(O)n2)=O)C)ccc([N+](=O)[O-])cc1 N1(C(c2ccc(C)o2)=O)CCN(C(=O)Cc2cnn(C(C)C)c2)C(CC2CC2)C1 C1(C(N(CCC(c2cccs2)NC(=O)C2=CCSC2)C)=O)CCC2CC1CO2 N(C1c2ccccc2OCC1F)C(=O)NCc1ccc(OCCC)cc1 Cc1c(C(=O)NCCCNC(=O)COCC2CCCC2)ccc(F)c1F N1(C(c2cc(C(C)C)n(C)n2)=O)C(CNC(=O)COC2COC2)CC2COCC12 c1(C(N2C(CNC(C(C=CC)O)=O)CC(O)C2)=O)cc(C)nc2c1CCCC2 C(CC)(CCCC(=O)NC(C)C(C)C(=O)OC)NC(c1n(CC#C)ccc1)=O c1(C(c2n(CC)nnn2)NCc2cc(C(=O)OC)no2)c(F)cc(Cl)cc1F Cc1cc(C(=O)NC2CCC2NC(c2ccc(C)n2C)=O)c2c(O)nn(C)c2n1 C12(C(=O)NC(C3(O)CCN(C(=O)CC4CC(C)(C)CO4)C3)C)CC(C)(CO1)C2 c1(CNC(C2CC(=O)N(c3cccc(Br)c3)C2)=O)ccc([N+](=O)[O-])cc1Cl C1(C(C)NC(=O)CC(C)c2cnn(C)c2)CN(C(c2coc(Br)n2)=O)CCO1 C1(C(=O)NC(C2CCCN2C(c2ccc(=O)oc2)=O)(C)C)(OC)CCCOC1 C1(C(=O)NC(C(C(=O)NCC(C(C)C)CO)C)C)CCC(C2CC2)C1 N1(C(C)=O)CC(O)CC1C(=O)OCc1cc(Br)c(Br)o1 c1(OC)ccccc1C(C)=CC(=O)OC(c1cccc([N+](=O)[O-])c1)C C(=O)(C(O)CCNC(N)=O)N(C)Cc1onc(C)n1.N12CCCC1C2 Cc1nc2ccc(CNc3scnc3C(N)=O)cc2o1.N12CC(CC(F)C1)C2=O CCC(C(=O)OC)C(=O)NCCCCCC(=O)NCC1(COC)CCC(=O)N1 c1(C(N2CCN(C(CC3C(C)C3)=O)CC2C2CC2)=O)cnc2c(=O)[nH]ccc2c1 CCCCCC(F)C(=O)N1CC=C(C(=O)Nc2coc(OCC)n2)CC1 N1(C(CC(CCC)O)=O)CCC2(C1)CN(C(c1c[nH]nc1-c1ccncc1)=O)C2 c1(C(N(CCNC(CC(=C)C)=O)CC)=O)cc(N(C)C)cc(Br)c1 N1(C(c2c(CC)ncnc2)=O)CCCC(NC(c2cc(C(N)=O)cs2)=O)CCC1 N1(C(c2nc(C)c(Br)cc2)=O)CCC(NC(=O)C(=O)NCCC(C)C)C(C)(C)C1 C1(C(=O)NCC2(CNC(CCc3n(C)ccc3)=O)CC2)CCc2nnnn2C1 C1(NC(=O)CCN2CCCC2)CCCCC1CNC(c1scnc1Cl)=O C(=O)(C1CCc2nccn21)N(C1CCN(C(=O)Cc2cn[nH]c2)C1)CCO C1(C)(NC(CCNC(=O)OCC)=O)CCN(C(c2nccnc2OC)=O)C1 N1(C(c2cn(C)nn2)C)CC(n2cc(C3(O)CN(CC(C)(C)C)C3)nn2)C(C)C1 C#Cc1cnc(NCC(C)NC(c2c[nH]nc2-c2cccs2)=O)nc1 C12(NC(c3ccc(CNC(C)=O)o3)=O)CCOC(CNC(COCC=C)=O)(C1)C2 Cc1nc(NC2CN(C(=O)C(n3nc(C)cc3C)C)CC2(C)C)cc(Cl)n1 N1(C(C2C(C)=C2)=O)CC2(CCCC2NC(C2CCC(C)CC2)=O)C1 c1(C(=O)NC(C)CNC(=O)CC2CCCCO2)c(Cl)ccc([N+](=O)[O-])c1Cl CCCCCS(=O)(=O)CC(=O)N1CC(NC(=O)COCC(C)(C)C)C(C)C1 C1(C(=O)NC2CCC(OC)C2)CCN(C(C23CCCN2CCC3)=O)C(C)(C)C1 C1(C(N(CCSC)CC)=O)N(C(=O)C(CSC)OC)CCC1(C)C c1(NC(C2C(CC)CCN2C(c2ccnc(OC)n2)=O)=O)ccc(O)c(F)c1 O(N=C(CN(C1(C(=O)OC)CNC1)C)c1ccccc1)CC CC1(CNC(c2ccc(CO)cc2)=O)CCCN(C(C2OC3CCC2CC3)=O)C1 CCC(C)(O)CCNC(=O)CC(C)N(C)C(c1csnc1C)=O Cn1cc(C(N2CCCC2(C)C(=O)NCCC(O)CCO)=O)ncc1=O c1(C(=O)OCC)cc(C)n(CC(=O)NC2CCC(C)(C(=O)O)CC2)c1C c1(C(=O)NCC2N(C(c3nnn(CC)c3C)=O)CCC2)cccc([N+](=O)[O-])c1C C12(NC(C(C)NC(C)=O)=O)CCOCC1CN(C(c1cccn1C1CC1)=O)C2 C=CC1COCC1NC(C1(OC)CCN(C(c2cc(Cl)c[nH]2)=O)C1)=O c1(C(=O)NCC2C(NC(c3c(C)cco3)=O)C2)ccc(C(O)CF)cc1 N1(C(C(C)C2CCC2)=O)CC23CCCC2(C1)CN(C(=O)C=Cc1ccccc1)C3 c1(C(C(=O)N(CC(C)O)CCNC(c2cc[nH]n2)=O)C)ccc(Br)cc1 N1(C(C(=Cc2ccccc2)OC)=O)C2CCC1CN(C(=O)CCC(C)O)CC2 N1(C(c2ncc(Br)s2)C(=O)NCC2CCCO2)CCC(CC(F)F)(CO)CC1 C=CC(C)(C)CC(=O)NC1CC=CCC1C(=O)NCc1cccc(OC)c1 c1(N(C)C)ccc(CCC(=O)NC2CN(C(=O)CCc3cnco3)C2)cn1 c1(C(C)C)nnc(C=CC(=O)NCCC(C(C)C)NC(=O)CC2COC(=O)C2)o1 C(CC(F)F)(C(=O)NCC1(O)CC(O)C1)N(C(=O)CCC1CCOCC1)C C=C=CC(C)C(=O)NCCCN(C)C(C1CC2CCC1C2)=O N1(C(c2ccccn2)Cc2cccc(CCSC)c2)CCC2(CC1)OCCO2 C1(C(=O)NC(CC#C)CC(F)F)CC2CN(C(C3(OC)CCC(C)C3)=O)CC2C1 C(=O)(C(C)(C)CC(=O)NC1(CNC(=O)C(C)(C)c2ccn(C)n2)CCCC1)OC N1(C(Cc2ccc(C)o2)=O)CC2(CC2)CC1C(=O)NCC1(O)CCC(C)(C)C1 c1(C(=O)NCc2c(C(=O)NC(C)CC3CCOCC3)occ2)cc[n+]([O-])cc1 c1(NC)cccc(C(=O)NCCCC2CCN(C(c3[nH]cnc3C)=O)CC2)n1 C#Cc1ccc(C(=O)NC2(CNC(c3ccon3)=O)CCCCC2)cc1Cl CC(CN(C(=O)C(C1CCOCC1)C)C)C(=O)NCCCN1CCOCC1 c1(C(=O)NC(C2(CNC(c3occ4c3CCC4)=O)CC2)C)cnn2c1OCC2 C1(C(=O)OC)CC12CCCN(C(c1c(Cl)cc(OC(F)(F)F)cc1Br)=O)C2 N1(C(c2cc(C)sc2C)=O)CCCCC(C(N2CCC(OC(C)C)C2)=O)C1 C#Cc1cccc(C(N2CC(NC(C3(C)CC3)=O)CC(C)C2)=O)c1Cl C1(CNC(=O)CC2(O)CCCC2)CCCC(NC(c2cccc(C3CC3)c2)=O)C1 N1(C(C(C)NC(C)=O)=O)CCC2(CCN(c3nc(C(C)C)ncc3COC)C2)C1 c1(COC)ccc(C(N2CCCC(CNC(c3ccc(OC)nn3)=O)C2)=O)cc1 C1(C(=O)NCCCC(C)NC(=O)COCc2ccncc2)(COC)CC=CCC1 c1(C(N2CC(NC(c3ccc(C)c(CO)c3)=O)C(C)C2)=O)nc2ccccc2s1 C12(C(=O)NCC(CC#C)(C)C)CCN(C(c3csc(CO)n3)=O)CCC1C2 N1(C(CCNS(C)(=O)=O)=O)CC2CCC1CN2C(C1(CC2CC2)CC1)=O Cc1cc(=O)c(C(=O)NC(C2CCN(C(C3CCC3(C)C)=O)C2)C)cn1C1CC1 N1(CCC)CC(C(N2CCCC(N(C)Cc3ncc(C(C)(C)C)o3)C2)=O)CC1=O c1(CC)nc[nH]c1C(N1CC(=C(F)CNC(=O)C(CO)N(C)C)C1)=O C(=O)(CC(C)(C)C(=O)NCCCC(C)NC(C12CC=CC(C1)OC2)=O)OC N1(C(C2CC(SC)C2)=O)CC(NC(C2(O)CCSC2)=O)C(n2ccnn2)C1 C1(NC(C2CCc3nncn3C2)=O)CC2(CCCN(C(c3cnc(Cl)s3)=O)C2)C1 N1(C(Cc2c(C)nc[nH]2)=O)CCC2CCCC(C1)N2C(c1cn(C)cn1)=O c1(NC(C2CCN(C(C3CCc4nc[nH]c4C3)=O)C2)=O)ccc2cnccc2c1 CC1(C)C(CNC(c2coc(C3CCCCC3)n2)=O)CCN1C(c1ccsn1)=O CCCC(CC)CCC(=O)NC(C1(CNC(C2(O)CCC(C)(C)CC2)=O)CC1)C c1(CNC(C(CCC)(C)O)=O)ccc2c(c1)CCCC2NC(=O)C=CCOC CC1(CNC(=O)COC2CCCCCC2)CCCN1C(=O)Cn1ccc(C(F)F)n1 N1(C(CCC2C(C)C2)=O)C2CCC1CC(CNC(c1cccc(CO)n1)=O)C2 c1(N(CCC(N)=O)C)ccc(S(=O)(=O)N2CCOC3CCOCC23)cc1C#N C(=O)(C(O)C(F)(F)F)NC(C1CCN(C(C(C2CCOCC2)C)=O)CC1)(C)C c1(CC(C)N(C)C(=O)Nc2ccc(-n3cnnn3)cc2)cccc(F)c1 C1(OCc2cn(Cc3nc(C)sc3)nn2)CCCC(NC(c2ncccc2N)=O)C1 C1(N(C(c2scc(C)c2)=O)CC2CC2)CCN(C(c2ccnn2CC2CC2)=O)CC1 N1(C(CC(=C)C)=O)CCC(N(CC(C)C)C(=O)CC2C=CS(=O)(=O)C2)CC1 c1(C(=O)NCC2N(Cc3ccnc(SC)n3)CC2)cc2ncccc2s1 C1(CC)CCCCC1O.c12nc(cs1)C(=O)NOCC(=O)NC2 CC(CC(=O)NCCCC1CN(C(=O)CS(N)(=O)=O)CCO1)C(F)(F)F c1(C(=O)OCC(c2ccc(C(CC)C)cc2)=O)cc(=O)n(C)cc1Br C1(C(N2C3(CNC(c4nc(C(C)(C)C)oc4)=O)CC(C2)C3)=O)COC2COCC12 CN1CCCCC1CNC(=O)C(O)CNC(C1(O)CCCCC1)=O C(=O)(C1c2c[nH]nc2CCC1C)N(CCNC(CCC=C)=O)CC1CC1 c1(C(CNC(=O)CC2CN(C)C2)NC(C2(CC#C)CCC2)=O)ccc(C)cc1 C1(NC(C2N(C(C)C)C(=O)CC2)=O)COC2(C1)CN(C(c1cncc(N)n1)=O)C2 c1(C(N2CCC(C(F)F)(CNC(C(C)OCC)=O)C2)=O)c(Cl)nc2sc(C)cn12 C1(CNC(CCC(=O)OC(C)(C)C)=O)CN(C(c2ccoc2)=O)CC1(F)CO N1(C(C(C)=C2CC2)=O)CC(CNC(C2(CO)CCOCC2)=O)OC(C(F)(F)F)C1 N1(C(c2ccc(CNC(c3c(CC)csc3)=O)nc2)=O)CCCC12CCNC2=O c1(COC(C2(c3cn(C)nc3)CCCO2)=O)cc([N+](=O)[O-])c(Cl)c([N+](=O)[O-])c1 c1(C(N2CCC(N(C(=O)CC3CCCC3)C)C2)=O)ccc(C#N)o1 N1(C(c2ccc(F)c(C)c2O)=O)CCN(C(C2CCN(C)C2C)=O)CC(C)(F)C1 Cn1c(C(=O)NC2CCCCC2NC(=O)C(c2cccnc2)O)cnc1O C1(CNC(C2CC3(CCC3)CO2)=O)CC2COCC2N1C(C12CCC(C1)OC2)=O C(CC)(C(=O)NC(C1CCCCC1)CNC(c1cscc1OC)=O)OCC C(=O)(CCCCCF)N1CCCC(CC(=O)NC(c2n[nH]c(C3CC3)n2)C)C1 c1(NC(C2N(Cc3ccc(C)c(Br)c3)CC(O)C2)=O)c(C)cc(F)cc1Cl c1(CC(=O)NCC(C2(O)CCN(C(c3c(C)ocn3)=O)C2)C)cccc(F)c1F C1(NC(C(C(CC)C)O)=O)CN(C(=O)C(C)C2CC2)CC12CCOCC2 C1(O)(CNC(CC2CCN(C)C2)=O)CCN(C(=O)CCCC2CCC2)C1 C=CCC(C)(CC=C)NC(C12CC(NC(=O)C(F)n3ccnc3)(C1)C2)=O c1(C(N(C)CC2N(C(C(C)=C3CCC3)=O)CCC2)=O)cc(C#N)no1 c1(OC)cccc(Br)c1C(=O)NC(CNC(=O)C1=COCCO1)C(C)(C)C c1(C(=O)OCC)n[nH]c(=NCCC2CC(NC(C3CSC3)=O)C2)s1 c1(OCC(=O)NCCCC(C)NC(C2(O)CCSC2)=O)cc(F)cc(F)c1 CC1CCC(CNC(C2CC(n3ccnc3)C2)=O)N(C(=O)C=Cc2cc[nH]n2)C1 CCCCC(C(=O)N1CC(CC(C)NC(=O)OC(C)(C)C)C1)N(c1ccon1)C N1(C(C(CC)CCOC)=O)CC(NC(=O)Cc2cscn2)C2CCCCC12 N1(C(c2c(C#C)c[nH]n2)=O)CC(C)C(NC(c2cscc2Br)=O)C(C)C1 Nc1ccc(S(=O)(=O)NC(c2cn3ccc(Br)cc3n2)=O)cc1Br c1(C(N2CCC(CNC(C=NOC)=O)CC2)=O)cc2scnc2[nH]1 C1(NC(CC2CCN(C(C(C)OCCCC)=O)CC2)=O)C(=O)NCC1(C)C C(=O)(C(C(C)(C)C)OC)NCC(CO)NC(c1cn(CCC)nn1)=O N1(C(CC(CC)SC)=O)CCCCC(NC(c2ncccc2Cl)=O)C1 C1(NC(=O)COC2CC2(F)F)CCC2(CC1)CCN(C(=O)COCC1CC1)C2 C#CC1(C(=O)NCc2cnns2)CCN(C(=O)CN2CC3CC3C2)CC1 n1(CCC)ncc(C(=O)NCC2CCCC2NC(C2CCCS2(=O)=O)=O)c1C Cc1cc(=NC(CCF)C2CCCCC2)[nH]c(N2CCC(CS(C)(=O)=O)CC2)n1 C1(C(=O)NCC(CCCC)NC(=O)C(C)(C)C(C)C)CCC2(CCC2)CC1 c1(C(N2CC3CC(C(N4C(CC=C)CCCC4)=O)(C2)C3)=O)nccc2[nH]ccc12 N1(C(c2c(C)[nH]cc2)=O)CCOC2(CCCN(C(C3CC(C(C)C)C3)=O)C2)C1 c1(N2CCC(CNC(C3CC(CC)OCC3)=O)CC2)nc2ccc(F)cc2o1 C1(C(=O)NCC(c2ccc(F)cc2F)CO)Cc2cc(Cl)ccc2O1 C=CC(O)C(=O)NCCCN(CCCNC(c1coc(C(C)OC)n1)=O)C c1(NC(c2n(CCC)nnn2)c2nc(C(F)(F)F)cs2)ccc(F)c(CO)c1 C1(C(=O)OC)CCCN(C(C2CCN2C(c2ccc(Cl)cc2)=O)=O)C1 c1(NC(C(COC)NC(=O)Cc2cncs2)=O)ccccc1CCO C1(C)(CNC(CC2ON=C(C)C2)=O)CCN(C(C2(F)CCOC2C)=O)CC1 N(C1CCc2cc(F)c(F)c(F)c21)CCOc1cc(C)c(F)cc1F C=CC1COCCN1C(=O)CC1(C)CCN(C(=O)C(CCC)=CCC)C1 c1(CC(N2C(C)C(NC(=O)CC3CC3)CC2)=O)cc2ccccc2nc1O c1(N2C(C)CC(NC(c3cccc4ncoc34)=O)CC2)ncnc(Cl)c1[N+](=O)[O-] N1(C(c2cccnc2CNC(=O)C2=C(C)OCCS2)=O)CCC2CCCC12.CO c1(C(=O)NC23C(CN(C(C(CC#C)(C)CC)=O)C2)C3)cnn2ccc(Cl)c(F)c12 N1(C(C2CCC(C)C2)=O)CCC2(CC1)CCN(C(c1cnn3ccccc13)=O)C2 N1(C(c2c(C)ccc(O)c2)=O)CC(C)N(C(c2cc(C3CC3)n(C)n2)=O)CC1C Cc1nnsc1C(=O)NCC1(CC2CC2NC2(c3ccccc3)CC2(F)F)CC1 C1(N(C)C(C2CCC(F)C2)=O)CCC(NC(=O)CCOC2CCOCC2)CC1 C1(CC)CCCN2C(=O)N(CCCCCC3CC3)C(=O)C2C1 Cc1cc2c(cc1NC(=O)NC(C)C(O)C(F)F)CCO2 N1(C(C=CC)=O)CCC2CCN(C(c3ccc(C)s3)=O)C2C1 N1(C(C2(C(C)C)CCC2)=O)CCN(C(=O)C(N)=O)C(CC(F)F)C1 C1(C)(CC)CC(C(=O)NCC2CN(C(=O)CCCF)CC2(C)C)CCO1 C(CC(C)C(=O)NCCOCCCN(C(=O)CSc1nccn1C)C)OC O=C1Cc2c(C(N3CCCC3C(N3Cc4cc(Br)cnc4C3)=O)=O)cccc2N1 CCC(C)CC(=O)N(C)CC1CCCCN1C(=O)C=CCN1CCC1 C(=O)(C1=C(C)OCC1)NC1(CNC(CCOC(C)=O)=O)CCC1 c1(C(=O)Nc2csc(-c3cccc([N+](=O)[O-])c3)n2)nnc2n1CCC(C(F)(F)F)C2 CC(c1ccc(F)cc1F)=CC(=O)NC(C)C(C)NC(=O)CCc1ccc(C)s1 CCCC(CCC)C(=O)N1CC2C(NC(c3nc(Cl)ccc3F)=O)C2C1 c1(C(=O)NCC2CCC(NC(C3(C)ON=C(C)C3)=O)C2)c(C)cc(O)nc1C C1(C(=O)NCC2CCN(C(=O)CCc3cscn3)C2)COc2ccc(Cl)cc2C1 CC1CNC(=O)CN1C(C1C=CCN1C(=O)CC(F)(F)F)=O C1(CNC(C(CCC)OC)=O)CC2(CO1)CN(C(=O)CCCC(OC)OC)C2 C(CCCCNC(C)=O)N(C1(C(=O)NC(=O)C(O)CC2CCCC2)CC1)C(C)C N1(C(Cc2c(C)nc[nH]2)=O)CC(C)CN(C(C2CC3CCCCN3C2)=O)C(C)C1 C1(OCc2cc(C(=O)OC)n[nH]2)CN(C(=O)COC2CCCC2)CC(F)(F)C1 c1(CC)ccc(CSc2nnc(-c3ccc(C)o3)n2CC2CC2)n1C.N Cc1ccc(S(=O)(=O)NCC2COCCN2C(c2cc(F)c(F)cc2O)=O)cn1 c1(CC(=O)NC2CC(C)(NC(c3cc(C)cc(F)c3)=O)C2)ccccc1[N+](=O)[O-] N1(C(C(C2CC(NC(c3occc3C3CC3)=O)C2)F)=O)CCC2(CC1)N=N2 Cc1cc([N+](=O)[O-])ccc1C(=O)NCC(C)CNC(=O)CCc1ccc(F)nc1 C1(CNC(CN(CC(=O)NC(C)C)C)=O)CN(C)CCN1C(C1CCCO1)=O C(=O)(C1=NNC(=O)CC1)N1CCC(N(C(=O)C2=CCCS2)CCC)C1 CCC(CC)(CC)C(C(=O)N1CC(C(=O)OC)C(C)C1)OC O(NC(=O)CC(O)CNC(C1CC2(CC2)CN1C)=O)CC(C)O Cn1nnc(C(=O)NC2C3CC(NC(C4CC(F)(F)C4)=O)CC23)c1N CC(C)CC(C)(CNC(c1cc(C(F)F)[nH]n1)=O)NC(c1cc(Cl)c(Cl)[nH]1)=O C(=O)(CC1CCCc2ccccc21)N1CCCCC(NC(C2CC3CC2C3)=O)C1 C12CCN(CC1)C(=O)C(CO)NC2C.C1(C(=O)NC(N)=O)CC1C(F)(F)F c1(C(N)=O)n[nH]c(=NC2CN(C(c3cnc4n3CCCC4)=O)CC23CCC3)s1 n1(CC(=O)N(C2CCC(NC(=O)CO)C2)C)cnc2ccc(F)cc2c1=O C1(OC)CC(NC(=O)CCc2ccc(Cl)cc2Cl)CN(C(c2cc(C)co2)=O)C1 C1(CNC(C(N)=O)=O)(CO)CC12CCN(C(c1csc(Cl)n1)=O)CC2 CC(C)C(C(=O)NCC(O)CNC(=O)CCN1CCOCC1)NC(=O)C(F)(F)F C1(N(C(CNC(CN(C)C)=O)=O)C)CCCCN(C(=O)Cc2ccccc2O)C1 CC(C)CC(C(=O)N1CC(NC(=O)COC2CC2)C1)NC(=O)Oc1ccccn1 CCCCS(=O)(=O)CC(=O)NCC1CC2CCC1N(C(=O)C1=CCSC1)C2 C1(NC(c2cnn(CC)n2)=O)CCN(C(c2cc(C)ccc2OC)=O)C12CCC2 C1(NC(C2C(C)OCC2)=O)Cc2ccccc2N(C(C2CCCN2C=O)=O)C1 c1(OC)ccc(F)cc1CC1CC(CCNc2ncc(F)cn2)C1 CC1(c2cn(C3CC(N(C(=O)CCCC4CCC4)n4cccn4)C3)nn2)CCOC1 CCCC(CNC(=O)C(C)S(N)(=O)=O)C(=O)NCc1ncccc1Cl c1(C(=O)OC)ccc(C(N2CCCCC2CNC2CCC2)C(=O)NC2CC2)nc1 C1(OC)(CNC(C23CCC2CC3)=O)CN(C(=O)CSc2nncn2C)C1 c1(OC)ccc(C(N2CCN(C(c3cnc(Cl)cc3Cl)=O)C(CO)C2)=O)nc1Cl c1(CNC(C2CCCN2c2cc3ncnn3cn2)=O)c(F)cc(Cl)cc1Cl C1(CNC(C(CCC)O)=O)CN(C(=O)CN2CCOCC2)CCC1C(F)(F)F c1(NC(C(CCOCCO)NC(=O)CC2(O)CCC2)=O)cnc2[nH]cnc2c1 c1(CN2CC(C)(c3cn(-c4ccc(Cl)cc4F)nn3)C2)cc(I)ccc1[N+](=O)[O-] C1(C)(C(=O)NCC(N(OC)C)=O)CCCN(C(c2cc(C)n(C)c2C)=O)C1 CCCN(OC)C(=O)CC1CC(C)N(C(=O)C(O)C2CCC2)C1 C=CC(C)(CCOC)C(=O)NCCC(O)CNC(c1cnoc1C)=O c1(C(=O)NCC2CN(C(Cn3nnc(=N)[nH]3)=O)CC2(F)F)cccn2nnnc12 c1(CC)cc(F)ccc1C(=O)N(CCCN(C(=O)CCNC(=O)CO)C)C c1(C(N)=O)cc(C(=O)NC2CC(F)(CNC(=O)Cc3csc(Cl)n3)C2)on1 c1(C(N2C(CNC(C3(C)CC3(Cl)Cl)=O)C=CC2)=O)cccc([N+](=O)[O-])c1N c1(C(C(=O)N(C2CCCCC2)CCNC(c2nnc(C)s2)=O)C)c(C)n[nH]c1C C(c1csc2ccccc12)=CC(N1C(CNC(C2CC(N(C)C)C2)=O)CCC1)=O c1(NC(CN2C(CCNC(CCC=C)=O)CCC2)=O)ccc(NC(C)=O)cc1 c1(OC)ccc(C(N2CC(NC(c3cc(C4CC4)on3)=O)CC(O)C2)=O)cc1C C(=O)(C(CC)C(=O)N1CCC1CC(N1CC2CC1CS2)=O)OCC CC1CC(NC(=O)CCNC(N)=O)CN1C(=O)CCOc1cccc(Br)c1 Cc1cccnc1C(F)(F)C(=O)NC(Cc1ccc(Cl)cc1)CC(=O)O Cc1cc(CC(=O)NC(C)C(=O)NCc2noc(C3CC3)n2)cs1 Cc1cc(CNC(C2CCN(C(=O)C3=NOC(C)C3)C23CC3)=O)ccc1O N1(CC(COC)O)CCN(C(=O)CC(C)OC(c2ccc(OC)cc2)=O)CC1 c1(C(C=O)=O)c(F)cccc1Cl.n1(C2CNC2)cc(-c2c[nH]nc2F)nn1 c1(C(=O)Nc2onc3ccccc23)ccc2c(C3=CCOCC3)cccc2c1 c1(C(=O)NC(C(C)C)(C)CNC(=O)CC2(C)CCC2)ccc(C(C)(C)C)c(Cl)c1 C(=O)(C1=C(Cl)CCOC1)N1C(CNC(=O)C=CBr)C2CCC1C2 C(CC(=O)N1CC2CC(O)CC2C1)(C(C)(C)C)NC(C(CC)C)=O C1(CC)NC(=O)N(c2cccc(CSc3cc(C4OCCO4)on3)c2)C1=O CC1CN(C(c2sccc2Cl)=O)CCC1N=c1[nH]n(C)cc1[N+](=O)[O-] C(CC(C)C)(C(c1nnnn1CC1CCOCC1)NCCC1CC1)OC c1(NC(c2cccc(SC(F)(F)F)c2)=O)ccc(Cl)cc1SC(F)(F)F N1(C(C2C(=C)CC2)=O)CC(F)CC1CNC(=O)COc1ccc(Br)cn1 c1(C(=O)NC2CCN(C(C3CCC(CC)C3)=O)CC2)cncc2c[nH]nc12 C=C(C)CCCC(=O)NC(CNC(=O)Cc1c(C)cnn1C)CC(F)(F)F CC1=NOC2(C1)CC(C(N1CC3(C1)SCCC3NC(c1cnn[nH]1)=O)=O)C2 S(=O)(=O)(c1ccc2c(c1)CC(=O)N2C)NCC(C(=O)OC)C.C1(=O)C(C)N1C(C)=O c1(C(N(CCCNC(C2C(SC)CCC2)=O)C)=O)c(C)nn(C)c1C(F)F N1(C(C2CCCN(C(CCCS(N)(=O)=O)=O)C2)=O)CCC2(CCC(=O)N2)CC1 c1(CNC(C2(C)CNC(=O)C2)=O)cnn2c1CN(C(=O)C(O)C1CC1)CC2 N1(C(Cn2cnc(C#N)n2)=O)CCCC(C2CCCN(C(=O)C3=CCCS3)C2)C1 C(=O)(C1CCCc2scnc21)N(C1CN(C(C2CCC(=O)NC2)=O)C1)C C(=O)(CC(C)(C)C(F)F)N1CCN(C(CC(CCC)C)=O)CC1CO c1(C(N2CC(C(Cn3cc(COCC)nn3)F)C2)=O)ccc(SC(C)(C)C)nc1 N1(C(c2ccnc(C(C)C)n2)=O)CC2(COC(CNC(C3CC3F)=O)C2)C1 c1(C(=O)NCC(C2CC2)NC(C(C)(O)CC(F)F)=O)cc2c(nc1O)CCC2 c1(-c2ccc(SC)nc2)n[nH]c2cccc(C(=O)NCC3COC3)c12 c1(OC)ccc(NCC(=O)NC2CC(CNC(=O)C(F)C3CCOC3)C2)cn1 c1(C(C)C)ncc(C(=O)N(CCCOCCNC(=O)C(F)C2CCC2)C)s1 C1(C(N2CCC(O)(CNC(Cn3ccc(C)n3)=O)CC2)=O)CCS(=O)(=O)C(C)C1 Cc1cc(C(=O)NC2C3CCN(C(=O)CCS(C)(=O)=O)C23)cc(C)c1F C1(CN(CC)Cc2ccc(-c3nc[nH]n3)cc2)CCCCN1C(=O)OC(C)(C)C Cc1ccccc1C=CC(N1CCC(C(C)NC(c2cccnn2)=O)CC1)=O CC1(C)CN(CC2CCCC2)CCC1NC(=O)Cc1ccc(Cl)cn1 N1(CCCc2ccc(C)s2)CCOC(CNC(=O)Cc2nocc2C)C1 C1(NC(CCOCC#C)=O)CN(c2ncc(CC)cn2)CC2(CCC2)C1 N1(C(Cc2nc(=N)[nH][nH]2)=O)CCC(CNC(C2(F)CCCC2)=O)C12CCC2 Nc1ccc(C(=O)NC2CC2CNC(c2ccc(Cl)cn2)=O)c2ccncc12 c1(C(=O)NC(CC)CN(C(=O)CCC(=O)N(C)C)C)cc(Br)cnc1S n1(CC)ccc2nc(N3CCC3C(=O)NCCOc3ccccc3Cl)ncc12 C1(C(=O)NCc2c[nH]cc2C2CC2)CCCCCN1C(=O)CC1CCCCN1C N1(C(CCC(=O)NC)=O)CC2(C)CC1C2NC(=O)CC1SC(=N)NC1=O Cc1nc2ccc(C(N3CCC(CCNC(C4COC(C)(C)O4)=O)C3)=O)cn2n1 C1(C)(C(N2CCC(C(C)NC(C=Cc3c(C)n[nH]c3)=O)CC2)=O)CCN(C)C1=O C#CCC(C(N)=O)NC(c1cnc(CNC(=O)C(C)=CC(C)(C)C)nc1)=O C1(C(=O)NCC23N(C(c4nnsc4C)=O)CC(CC)(C2)C3)CN2CCCN1CC2 C(C(=O)NCCCN(C(=O)CC1CCCCC1O)C(C)C)(C(C)C)N(CC)CC Cc1ccnc(C(=O)NC(CC2CCOCC2)C(=O)NCC(=O)Nc2cccs2)c1 n1(C(C)C)ncc(C(=O)NCC2CCN(C(=O)Cc3cc(C4CC4)no3)C2)c1N c1(CNC(C)=O)ccc2c(c1)CCC2NC(c1cnn(C(C)C)n1)=O C12(C(N3CCC(CCC)C3)=O)CCN(C1)C2.c1(SC)oc(C)nc1C CC1CC(C(N2CC(C(C)NC(=O)CN(CC(=O)N(C)C3CC3)C)C2)=O)CCS1 N1(C(C2C(C)OCCO2)=O)CCN(C(c2cn(CC(N)=O)nn2)=O)CCC1C CC1C(NC(c2coc(C(F)F)c2)=O)CCCN1C(=O)C=Cc1cc[nH]n1 CC1(C)CCc2cc(CN3CCOC(c4cccc(C#N)c4)C3)ccc21 C1(NC(C(CC)OCC)=O)CN(C(c2nnc(C)s2)=O)CC1C N1(C(Cc2cc(OC)ncc2)=O)CC(NC(=O)CCc2n[nH]c(=N)s2)C(C)(C)C1 C(=O)(C1=CCCC1(C)C)N1CCN(C(c2ccc(C(C)(F)F)cn2)=O)CC1CO Cc1nc(C#N)cc(=NCC2CC(C)N(C(=O)CCc3cccs3)C2)[nH]1 C1(NC(c2c(C)nsc2)=O)(CF)CCN(C(C2C(C)(C)C2(F)F)=O)C1 c1(C(NC(NCc2cccc(OCC)c2)=NC)C)c[nH]c2cccc(F)c12 Cc1nc(NCCC(C)NC(C2CCCCC2)=O)c2ccsc2n1 c1(NC(C2NCCN(C(Cc3ccc(C)nc3)=O)C2)=O)ccc(I)cc1[N+](=O)[O-] N1(C(CCC)=O)CCC(C(=O)Nc2ccc(C3SCCCS3)cc2)CC1 O=S(=O)(c1cc(Br)c(O)c(Br)c1)NCC1CC1CO c1(C(N2CC(N(C(C(C(=O)OCC)CC)=O)C)C2)=O)csc2cc(OC)ccc12 CS(=O)c1ccccc1-c1nc(C(=O)Nc2ccc3[nH]ccc3n2)cs1 CCC(C)C(O)C(=O)NCC1(C(=O)NC(CCO)C(C)C)CC12CCC2 c1(C(c2n(CCC)nnn2)Nc2cccc(OC3CC3)c2)c(C)nn(C)c1C C(c1ccc(CO)o1)=CC(N1CCC(CNC(=O)C(F)C2CCC2)C1)=O C1(CC=C)(NC(c2ccc[n+]([O-])c2)=O)CCN(C(=O)C(C)(C)n2cnnn2)C1 c1(C(N(CCNC(CC=C)=O)C2CC2)=O)cc(Br)c(C)s1 CN=c1ccc(C(N2CC3CC3C2C(=O)NCCCS(C)=O)=O)c[nH]1 C1(C(=O)NC2CC2CN(CC(=O)NC2CC2)C2CCC2)CCCO1 c1(SCC(=O)NCC2(O)CCN(C(C(C)CSC#N)=O)C2)ccc(F)cc1 C1(NC(CC(CC)C)=O)CCN(C(C2CCC(=O)C2)=O)C1(C)C C12(C(N3C(C(=O)NCC4CC(SC)C4)COCC3)=O)CCCN(CC1)C2 N1(CC)CCc2ccccc2C(CC(=O)OC)C1.c12nn(C)cc1NC2=O C(C(C)(C)CC(=O)N1CCCC(C(C)C)CC1)NC(C(C)OCCCC)=O c1(C(=O)NC(C#C)C)cc2cc(-c3sccc3CO)ccc2o1 CC1(C)CCCCC1C(=O)N(CCNC(=O)C(O)Cc1ccc(Cl)cc1)C1CC1 c1(N2CCCC(CCNC(c3nccc(CC)c3)=O)C2)cc(O)nc(=O)n1C N1(c2nccc(-c3n(C)ncc3)n2)CCCC2(CC(NC(C3CC3(C)C)=O)C2)C1 c1(OC)ccccc1N(C)C(c1ccccc1NC(c1ccc(Br)o1)=O)=O Cc1n[nH]c(C)c1CC(C)C(=O)NCCCN(C(C1CCC(F)CC1)=O)C1CC1 CCCC(CN=C(NCC1CC1)N1CCC(C)(c2ccccc2)CC1)OCC CCC(C)C(C(=O)NC1CCOCC1C)N(C)C(c1nnn(C)c1N)=O Cc1ccc2[nH]c(C(=O)NC(C)C(C)(C)NC(=O)CCOCC(F)(F)F)cc2c1 c1(C(=O)NC2CCC(CNC(CC3N(C)CC=CC3)=O)CC2)c(Cl)ccnc1F C(=O)(C(C)(C)c1ccn(C)n1)NCCOCCN(C)C(C1(CO)COC1)=O C(=O)(C(C)(C)S(=O)(=O)C1CC1)NC1CCCC(NC(CC(C)n2ccnc2)=O)C1 N1(C(C2CCC(CC)O2)=O)CCOCC(NC(=O)C=C(C)c2ccsc2)C1 N1(CCC)CC(C(=O)NCCCN(c2nnc(COC)s2)C)CC1=O N1(C(COCC(=O)OC)=O)CCC2CC2(C(N2CC(O)CC2CO)=O)CC1 C1(C(=O)NC(c2cccnc2)C)C2CCCC2CN1C(=O)COC1CC1 CC#CCCC(=O)N1CCCC1C1CCN(C(c2nnccc2C)=O)CC1 C1(CNCc2ccc(-c3ccc(-n4cc(C)c(C)n4)cc3)s2)CCC2(CCC2)C1 N1(C(C2C(C(=O)Nc3ncc(C)c(I)c3)C2)=O)CC2OCC(F)(F)C2C1 c1(C(=O)NCC2CCC(=O)NC2=O)nc2cccc(Cl)c2[nH]1 C1(CCOC)CN(C(=O)C(C)CC)CCN1C(=O)C(c1cccc(C)n1)(F)F C(C1=CCN(C(C2CN(C3COC3)C2)=O)CC1)NC(C(C)CN1CCOCC1)=O c1(C2(CN)CC2)ccccc1C(=O)NCC1(C2(O)CCCCC2)CC1 Cc1cc(Cl)cc(C(N2CC(NC(c3ccn(C)n3)=O)CC2C)=O)c1O N1(C(C2CN(CC)C(=O)C2)=O)CCN(C(c2ccnc(CO)c2)=O)C2CCCC12 N1(C(=O)Cc2ccoc2)CCCC(F)(C(=O)NC2CCCCC2F)C1 c1(C(N2CCN(C(C=C(C)C)=O)C(C)C2)=O)cnc2onc(C)c2c1 c1(OC)cccc2c1OCC(C(=O)NCC(CO)NC(=O)C1=NOC(C)C1)=C2 c1(C(=O)NCC#CCNC(C(c2cccc(F)c2)C)=O)ccc(O)c([N+](=O)[O-])c1 C(c1cc(F)c(F)c(F)c1)=CC(=O)OC.C1(CC(C)C)C(=O)N1C1CC2(CNC2)C1 c1(C(C)NC(N2CC(CNC(C(C)NC(C)=O)=O)C2)=O)noc(C)n1 c1(CC)cc(C(=O)NC2CCCC2NC(=O)C(CC)CC)nn1C C1(CNC(C(CC)(C)C)=O)CCCN(C(=O)C(O)Cc2ccccc2)CC1 CCCC(CCCNC(=O)C=C(C)c1ccccc1)NC(=O)COC(C)CC CC1CN(C(c2cc(F)cs2)=O)CC1NC(C1(Cc2ccccc2)CCC1)=O c1(C(=O)Nc2c(CC)noc2)cnc2ccc(Br)cc2c1Cl CCC(C)(C)C(O)C(=O)N1CCN(C(=O)C2=CC(C)(C)C2)CC1c1nccn1C N1(C(CCCCc2ccc(C)cc2)=O)CCCCC(NC(=O)C(O)C2CC2)CC1 CCC(F)(F)CC(=O)NC1CN(C(=O)C(C)NC(C)=O)CC1c1ccc(F)cc1 C1(C(=O)NC(C(=O)OCC)(C)C)CCCCCC1NC(C1CCC(=O)CC1)=O C1(NC(C(c2cnn(C)c2)C)=O)CC(C(=O)NCc2n[nH]cc2C)C1(C)C c1(C(=O)NC2CC3CC2N(C(C2CSC2)=O)C3)cc(F)c(CO)c(F)c1 n1(CC(=O)NC2(CCNC(CCC#C)=O)CCCC2)nc(Cl)ccc1=O C(CN(C)N1CCN(CC(C)(C)O)C(C(C)C)C1)c1cnc(C)s1 Cc1cc(CN2CC3CC(C2)N3C(=O)CNc2ncccn2)cc(O)c1 N1(C(C2C(C)C2)=O)CC2CCN(C(c3ccc(C(C4(C)CCCOC4)=O)[nH]3)=O)CC12 C1(C(=O)NC(CC)(C)CNC(=O)C(=O)N(C)C)CC2(C1)CC21CCC1 CCC1=NOC(C(N2CCC(C(=O)NCCOC(C)C)(CO)C2)=O)C1 C1(NC(CCC=C(C)C)=O)CC(C(=O)NC2CN(C)CC2(F)F)C12CCC2 Cn1ccc(C=CCCCCN2CCN(C(=O)OC(C)(C)C)CC2)c1 C1(NC(c2occ(C)c2C)=O)CN(C(=O)C(c2ccc(F)c(Cl)c2)O)CC1(C)C N1(C(C2CCN(C(=O)c3ccc[nH]3)O2)=O)CCCC2CCCCC12 C1(CNC(C=Cc2ncc(C)[nH]2)=O)CC(C)CN(C(=O)CCc2ccsc2Cl)C1 Cc1ccc(CC(N2CCC2C=Cc2cccs2)C(N2CCC(F)(C#N)C2)=O)c(O)c1 Cc1ncccc1-c1cn(CC(N2CCN(C(=O)C3=NOCC3)CC2)C2CCC2)nn1 C1(CC(=O)NCCC(c2cccc(Br)c2)O)CCC2(CC2)CO1 CN1CCC(C)(C(=O)NCCCC2CCCCN2C(=O)Cc2cnnn2C)CC1 C1(NC(=O)NCC(CC(=O)OC)C)C(C)(C)C(NC(=O)OC(C)(C)C)C1(C)C C(=O)(CC(C1CC1)NC(c1ncoc1C1CC1)=O)N1CC(C(C)OC)C1 C(C)(C(C)CC)(c1n(CC=C)nnn1)NCCCCc1cccs1 c1(C(=O)NCC(CN(C(c2c(C)nc(CC3CC3)o2)=O)C)O)cnc(Cl)c(N)c1 n1(CC(=O)NCC(CNC(c2ncc(CC)nc2)=O)C)ncn2cccc2c1=O c1(OC)ccc(CN2CC(C(=O)OCCOC(C)(C)C)OC(C)C2)nc1Cl N1(C(c2nc(N(C)C)oc2)=O)CC2CC(C(=O)NC34CCCCC3C4)(C2)C1 C1(C(=O)NCC2(CCC(=O)O)CC2(F)F)NCCOC12CCC2 C#CCC(CC(F)F)C(=O)N(C)CC1(O)CCN(C(=O)Cc2cnoc2)CC1 Cc1cc(NC(C2(C)CCCN(Cc3ccncc3Br)C2)=O)cc(Cl)c1 C1(CC(N2C(C(C)NC(=O)CN3CCOCC3)CCC2)=O)CC2CCC1C2 C1(CC(=O)OCC)CC2(C1)CC(F)(F)C2.N12CCN(C(=O)C1)C(=O)CC2 C1(C(N2CCCC(NC(C3(F)C4CCCC34)=O)C2)=O)CCS(=O)(=O)CC1 Cc1cc(C(=O)NC2CCC(NC(=O)CN3CCCCCC3)CC2)ncc1C#N C1(C(=O)NCCCN(C(CC2C(OC)CC2)=O)C)CCCC2(CCC2)C1 C12(NC(C3(COC)CC3)=O)CCC(CC1)N(C(c1cc(OC)n(C)n1)=O)C2 c1(NC)c(Cl)nc[nH]c1=NCCCCCCCCC(F)F CN1CCCC(O)(CC(=O)NCC2(C)CC(NC(c3cccc(Cl)c3N)=O)C2)C1 C(=O)(C1c2c[nH]nc2CN1C(=O)CC1CC(C2CC2)C1)NC(C(=O)OC)C C1(CCC(=O)NCCOC)CCCN1C(c1cnn(C)c1)=O c1(C(=O)NC2C(C)N(C(C3CC(C4CC4)=NO3)=O)CCC2)ccc2ncnn2c1 N1(C(C=CC(C)NC(=O)C=C2CCCCC2)=O)CCCCC1C1(O)CC1 C1(C(=O)NC(C(CO)NC(Cc2nc(C)oc2)=O)C)CCCCC1O c1(C(N2C(CNC(C3CC3C(F)F)=O)CC2)=O)ccc(CC2CC2)[nH]1 Cc1cc(F)c(C(N2CCC(CNC(=O)C(C)n3cnnn3)CC2)=O)cc1F CC1(C)CC(NC(C2CC(=O)CN2C(=O)C=Cc2ccncc2)=O)C12CCC2 c1(CCC)ccc(NC(C2(NC(=O)CCCn3ccnc3)CC2(C)C)=O)cc1 c1(C(N(C(C)CNC(=O)CCCC#N)CC)=O)cnc(C)c(C(=O)OC)c1 c1(CC(N2CCC(OCCNC(C3C(C)C3)=O)C2)=O)cccc(S(C)(=O)=O)c1 Cc1ccc2cccnc2c1C(=O)NCC1CC(F)(CNC(=O)CC(C)(F)F)C1 N1(CC)CCN(CC(N2CCOC(CNC(=O)C(C)C(C)O)C2)=O)C(=O)C1=O N1(C(C=C(COC)C)=O)CC2CC1CN(C(=O)CCCCCCSC)C2 CCCCC(CC)CC(=O)N1CC(C(=O)NCC(F)F)CC(C)C1 C1(NC(c2ccc(O)cc2Br)=O)CC12CCN(C(c1cccc(O)c1)=O)CC2 C=CC(C)(CCOC)C(=O)N1CC(O)CC1C(=O)NC(C)CN(C)C N1(C(COCC#C)=O)CCN(C(=O)C(C)N(C)C)C(C)C1 CC(CCCCO)NC(c1sccc1Cl)c1nnnn1C(C)(C)C c1(C(=O)NCCN(C2CCCC2)C(C2CC(CC)C2)=O)ccc2c(n1)CCOC2 C(=O)(C1=C(F)CN(C(c2nocc2C)=O)CC1)NC(C(=O)N(CC)CC)C C1(C)(NC(C2(F)CN(C(C3CCC(N(C)C)C3)=O)C2)=O)CCCC(C)(C)C1 CCCC(CCC)CC(=O)NCC(CO)NC(c1cnn2c1NCCC2)=O N1(CCC(=O)OC)CCCC(N(C(=O)CSc2nccn2C)C)C1 C1(C(=O)NC)C2CN(C(c3ccc(CNC(C4(C#N)CC4(C)C)=O)cn3)=O)CC12 c1(C(=O)NC2C=CC(C(=O)NCc3cccnc3)C2)cnc2ccc(F)cn12 c1(C(=O)NC2C(NC(C3(Cl)C(C)(C)C3)=O)CS(=O)(=O)C2)ccc(N)c([N+](=O)[O-])c1 c1(CC)nnc2c(C(=O)NCC3CCN(C(C4(CF)CC4(F)F)=O)C3)cccn12 C1(C(N2CCC(CC)C2)=O)CN(C(=O)C=Cc2cncs2)C2(CCC2)C1 c1(OC(C)C(N2CCCCC2CNC(=O)CN2CC3CC3C2)=O)ccc(F)cc1 C1(C(=O)NCC(C)OCC=C)N(C(=O)CC2CC(C3CC3)C2)CCCC1(C)C c1(C(=O)NC2CN(C(C(CC)C#N)=O)CC23CC3)cnc2c(Br)cccn12 c1(OC)cc(C(N2CCC(C)C(CNC(=O)C(O)C3CC3)C2)=O)ccc1[N+](=O)[O-] c1(C(N(C)CC2(O)CN(C(C(CC)N(CC)CC)=O)C2)=O)cc(F)c(C)cc1F C1(NC(C(C)C(F)F)=O)CN(C(c2cc([N+](=O)[O-])n[nH]2)=O)Cc2ccnn2C1 C1(OCC(=O)NCC(F)CNC(c2ccc[nH]2)=O)CCCC1 C#CC1CC2CCC1N(C(C1CCCC1CNC(c1cc(C)c(C)nn1)=O)=O)C2 c1(C(N2CC3(CN(C(C(n4c(C)ccn4)C)=O)C3)C2)=O)ccc(N=[N+]=[N-])cn1 C1(NC(C(C)OC(C)(C)C)=O)CCC(CC(=O)NCC2(O)CCN(C)C2)CC1 N1(C(CCCN(C(C)C)C)=O)CCN(CC(C)NC(=O)CC2CNC(=O)O2)CC1 C1(C(=O)NC(CC(=O)N(C(C)C(=O)O)C)C)CCN(C(c2ccccc2)C)CC1 C1(C(=O)NC(CCCNC(c2ncc(C)cc2C)=O)C)CC2COCC(C1)C2 NC(CC1CCCOC1)C(=O)Nc1nc(C2CCNCC2)cs1 c1(OC)cc(C(=O)NCC2(C(C)(C)O)CN(C(c3cccn3C)=O)C2)cnc1O Cc1cccc(C(=O)NCC(C2CC2)NC(=O)C(O)CC(N)=O)c1Br c1(C(N2CCC(NC(COCCOC)=O)C(F)C2)=O)cc2ccc(OC)cc2[nH]1 N1(C(c2c(CC)cno2)=O)CC2CC2(C(=O)NC2CCN(C(C)=O)C2)C1 N1(C(C2(C)CCC(=O)NC2)=O)CCC(C2CC2)(CNC(C2(O)COC2)=O)C1 c1(CC)c(C(N2CC3C(NC(C4CC(OC(F)(F)F)C4)=O)C3C2)=O)nnn1CC c1(C(=O)NCCCCCCNC(c2c(OC)c[nH]n2)=O)cc(S(N)(=O)=O)c[nH]1 CCCCCCCCS(=O)(=O)NCC1CCN(C(=O)CC(C)O)C1 C1([Si](C)(C)C)(CNC(C2(C)CN(C(C3C(OCC)CC3)=O)C2)=O)CC1 N1(C(CN(C(=O)C(F)(F)F)C)=O)CC2CC1CN2C(=O)CC1(C)CCS(=O)(=O)C1 Cc1ccc(F)c2oc(C(=O)NC3(CNC(c4cc(F)cnc4O)=O)CC3)cc12 c1(C(=O)NC2CCCC2NC(CSC)=O)cccc(NC(=O)CCc2cscn2)c1 c1(C(CC)NC(=O)NCC(C)OCC#C)cccc(S(=O)(=O)N(C)C)c1 C1(NC(c2c(C)oc(C(C)C)c2)=O)C2CC3CN(C(C4CC=CCC4)=O)C1C3C2 Cc1cc(C(C)NC(N2CC(C(=O)N(C)C)C2)=O)cc(F)c1 C1(N(C(C(CC)OC)=O)C)CCCCC1NC(c1sc(F)cc1C)=O C(=O)(CC1=CCOCC1)NCC(C)(C1CCC1)NC(CC(CC)C)=O Cc1cccc2cc(C(=O)NC3CCN(C(c4cc(F)n(C)n4)=O)C34CC4)oc12 c1(C(N2C(C(=O)NC3CCC4(CC4)C3)CSCC2)=O)ccc2[nH]ccc2n1 Cc1ccc(C=CC(N2CCN(C(=O)CCC(C)C)C(c3ncc[nH]3)C2)=O)cn1 C1(NC(c2c(C)occ2)=O)CC12CCC(NC(C1CC3C=CC1O3)=O)CC2 Cc1ccc(C)c(C(=O)NC2CC2CNC(=O)C(C)CF)n1 C1(CNC(C(F)OC)=O)CCC(F)(CNC(=O)C(O)CSC)CC1 N1(C(C#CC(CNC(C2CC(C)CC(C)C2)=O)(C)C)=O)CC2(CCCC2)CC1C N1(C(C(C=CCCC)O)=O)CCC(NC(C2(CCF)CC2)=O)C2(CCC2)C1 Cc1cc(=O)c(C(N2CC3CC3(NC(=O)CC3CC=CC3)C2)=O)cn1C n1(CCC)cc(C(=O)NCC2CCC(NC(=O)CN3CCOCC3)C2)nn1 N1(C(CC(CC)(F)F)=O)CCC2(CCC(NC(c3csc4nccn34)=O)C2)C1 N1(C(C2N(C(C)=O)CCOC2)=O)CCC2(CCN(C(=O)C(O)C3CC3)CC2)C1 c1(CCCC(=O)NCC2(COC)CN(C(=O)CC3(C)CC3F)C2)cccc(Cl)c1 CN1CC2CC(NCCc3cccc(Br)c3)CC(C2)C1 N1(C(c2cnc(CC)s2)=O)CCC2(CC1)CC2NC(C1CCC2CC1C2(C)C)=O N1(C(c2n(C)ncc2)=O)CCC2(CCCN(C(C3CC4(C3)CC43CCC3)=O)C2)C1 c1(C(C(=O)NC(CC)C)N(C(C)CC)CC)cc(C)c(C)cc1C c1(CC)cc(C(N2CCSC(CC)C2)C(=O)NCCCOC)ccn1 CCCC(C)(O)C(=O)NCCCCCN(C)C(c1cc(Cl)ccc1Cl)=O C1(C(F)(F)F)(NC(=O)NC(C(CC)(C)C)C)CCCC(C)(C)C1 N1(C(C(CC=C)(C)C)=O)CCN(C(c2ccc(OCCF)cc2)=O)CC(CO)C1 N1(C(c2c(CC)n(C)cc2)=O)CC2CCC1C1CN(C(C3CC3C3CC3)=O)CC21 C(=O)(C(F)C(C)(C)O)NCCOCCOCCCNC(CCC#C)=O N1(C(CC(C)(C)C#N)=O)CC2CCC(NC(C3CC4(CCOC4)C3)=O)CC2C1 C1(NC(C2CC(CNC(CCCNC(=O)OC)=O)C2)=O)CCN(C)CC1C CN1CCOC(C(=O)NC2CC(CCC(=O)NCCc3ccncn3)C2)C1 c1(C(=O)NCC(CO)NC(C2C=CCC2)=O)ccc2c(c1)CCCS2(=O)=O N#CC1(C2(O)CC(NCCc3cnn(-c4ccccc4)c3)C2)CCOCC1 C1(CNC(c2ccc(C)cn2)=O)CC(C(C)(C)C)CCN1C(=O)CCCC(F)F Cc1ccc2cc(C(=O)NC3CCCC(NC(c4ccc[nH]4)=O)C3)c(C)nc2c1 N1(C(CC(=O)NC)=O)CCCC2(CC(NC(c3cc(C(F)F)[nH]n3)=O)C2)C1 CC1CC(NC(=O)CSc2ccc(Cl)cc2)CCN1C(C1CCOCC1)=O C(C)(C)(CCC(=O)N1CCN(C(=O)CCc2ccccc2)CC1C)OC N1(C(c2ncc(C)nc2)=O)CCCC2C1CCN2C(c1c(Br)ccnc1Cl)=O c1(C2(C(N(CC(C)NC(=O)CC3(O)CC3)C)=O)CC2)cnn(C(C)(C)C)c1 CN1CCN(C(=O)NCC=C2CCNCC2)C(C2CC2)C1 C1(C(=O)NC(C(C)NC(COCCC(C)C)=O)(C)C)CC(c2ccccc2)=NO1 C1(C(=O)NCCCCN(CC)CC)COCCN1C(=O)CC1CC(C)C1 C1(C(=O)OC)CN(C(=O)C(N2CCCCC2CO)=O)CC1CC1C(=O)NN=C1C C1(C(C)C)CN(C(=O)CN(C)S(=O)(=O)N(C)C)CCN1C(=O)C(O)C(F)F C1(NC(C2CCOC2=O)=O)CCN(C(=O)C=CSCc2ccco2)CC1 C(=O)(C(C)(C(C)C)NC(c1cc(C(C)C)no1)=O)N1CCC(=C)CC1 C1(COC)COCCN1C(=O)C(C)(C)CNC(=O)Cc1ccns1 Cc1ncc(CC(=O)NC2CCC(CNC(C3C(C)(C)C3(F)F)=O)CC2)c(O)n1 Cc1cc(C(=O)NC2CCC(Cn3cc(C4(C)CC4)nn3)C2)c(C)s1 CCCCC(C(=O)N1CCC(CC)CC1)NC(=O)C=Cc1cncn1C CN(CCCC(=O)NC1CCCCCCC1NC(=O)C(C1CCCCC1)F)N=O N1(C(C(C)SCC)=O)Cc2n[nH]cc2C1C(=O)NCc1cc(C2CC2)n[nH]1 N1(C(c2ccc(C)c(Cl)c2)=O)CC(C)CN(C(c2cc[nH]c(=N)c2N)=O)CC1C N1(C(CCOCCN(C)C)=O)CCC2CCN(c3nc4ccccc4o3)CC2C1 C1(c2n(CC=C)nnn2)(Nc2ccc(C(=O)OCC)c(F)c2)CCC2COC1O2 C1(CNC(c2nc(C)sc2)=O)CCCCC1NC(=O)C(C1(O)CCCCC1)(F)F c1(C(=O)NCC(C)CNC(c2cnn[nH]2)=O)scnc1Br C(=O)(C1=CS(=O)CCC1)NC(C)CN(C)C(c1ncoc1C1CCCO1)=O CCC(CC)C(C)C(=O)N1CC(C)CCC1C(=O)NCC1CC2CCC1O2 c1(C2(C(=O)NC(CC)CNC(c3ncoc3C)=O)CC2)cccc(F)c1F N1(C(COCC)=O)CC2(C1)CN(C(c1cc[nH]c3nccc1-3)=O)CCO2 O=C(NNc1cccc(F)c1F)C12CSC(C1)C2 N1(CC(=O)N(C(C)(C)C)CC)CCN(CCn2nc(C)cc2C(F)(F)F)CC1=O N1(C(c2c(C)[nH]cc2)=O)CCC(NC(C2CC3CC3C2)=O)C12CC2 C1(NC(c2c(COC)cco2)=O)CC2(C1)CN(C(C1CC1Cl)=O)C2 c1(C(N2CC(CC)N(C(=O)C(C(C)CC)OC)CC2)=O)cc2c(nn1)OCCS2 c1(-n2c(-c3c(OCC)cccc3)nc(C)n2)ccc(Br)c(C)c1 N1(C(C2CCN(C)CC2)=O)CCOC2CN(C(=O)CN3CC4CC4C3)CC12 C1(C(N2CCN(C(C=CC=CCC)=O)CC2CCO)=O)CCc2cn(C)nc2C1 N1(c2nc(C)nc(-c3ccco3)c2)CC2CC1CN(C(C1CC1(F)F)=O)C2 C1(CNC(=O)Cc2cnoc2)CC(C(=O)NCc2csnn2)CO1 N1(C(c2ccc(SC)o2)=O)CCOCC1C(=O)NC(C(N)=O)C1CCCC1 CC1Oc2c(C(=O)N(CCCCNC(=O)C(C)(C)CF)C)cccc2NC1=O c1(CC(N2CCN(C(C(C)=C3CCCC3)=O)C3C2C3)=O)cc2ccccc2o1 C(C)(C)(CC(F)C(=O)NCc1nc(C)cs1)NC(CC(CC)C1CCC1)=O N1(C(C2OCC(C)(C)C2)=O)CCN(C(c2cnccn2)=O)C2CCCC12 c1(N(CCN(C)C)C)nc2cccnc2c(=NCCN(CCO)CCO)[nH]1 N1(CC(CCOC(C)C)O)C(C)Cc2cc(F)ccc2C1C c1(CC(=O)N(CCNC(=O)CCF)CC2CC2)ccc(Cl)cc1Cl S(=O)(=O)(CCC(=O)N1CCC(C(C)(C)NC(c2cncc(N)c2C)=O)C1)NC c1(C(C(=O)NCC2C(NC(COCCC=C)=O)C2)N(C)C)ccc(F)cc1 N1(C(=O)NC(c2ccc(Cl)cc2)(c2ccccc2)CC)CCC(OC)C(C)C1 c1(CCC)nc(C(=O)NCC2CCC(NC(C3(CS(N)(=O)=O)COC3)=O)C2)cs1 C1(Cc2onc(C(c3ccc(Cl)cc3)=O)n2)CCCC2(CCC2)C1 c1(N2CC(CCNC(C3CCC3(C)C)=O)(OC)C2)ccnc(S(C)(=O)=O)n1 CCCCCC(CC)C(=O)N1CC(CNC(C2CCOCC2(C)C)=O)C(C)C1 CC1CCC(C(=O)N(C)Cc2ncccn2)N(C(=O)C(F)CC2CCOC2)C1 c1(C(=O)NC2C(OC)CN(C(c3c(Cl)n[nH]c3C)=O)C2)nccc(N)c1Cl C1(NC(c2cc(O)cs2)=O)C=CCCC1C(N1CCCC(CO)C1)=O C1(NC(c2c(C)cco2)=O)CCCCC1NC(=O)CCc1ccccc1F C1(C(=O)NCC2C(C(=O)Nc3cn(CC)nc3C)CCC2)CCC(O)CN1C C(=O)(C(C)CC(C)(C)C)N1C(CC)C(C(=O)NC(CO)CCSC)CCC1 C1(C(=O)OC)(NC(=O)NCC2(Cl)CCCCC2)C2CCCC12 c1(OCC(=O)NCC23CC(NC(CCCC#C)=O)(C2)C3)cc(C)ccc1C(C)C CC(C)CC(CNC(c1ccc(=N)[nH]c1)=O)NC(c1ncccc1OC(F)F)=O c1(CC(CO)NC(C(c2ncccn2)C)=O)cccnc1F N1(C(C2(COC)CC2)=O)CCC2CCCC12CNC(c1ccc(C)c(C#N)c1)=O CC1CC(NC(c2ccc(CO)o2)=O)CN1C(c1sc(F)cc1Br)=O c1(C(=O)NCC(c2cnn(C)c2)NC(C(C)C2CC2)=O)ccc(C(O)CF)cc1 C=CCC(C(=O)N(C1CCCCN(C(=O)CNS(=O)(=O)N(C)C)C1)C)C(C)C C(=O)(C1CCc2cccc(O)c21)N1CCC(CNC(C(C)CC2CCC2)=O)CC1 N1(C(C2(C=C)CC2)=O)CC(CO)C2(C1)CN(C(C1(C(=O)OCC)CC3(CC3)C1)=O)C2 c1(NC(=O)Nc2ccc(C)nc2C)cc(Br)cc(F)c1O N1(C(CC=CC(C)(C)C)=O)CCC(CCNC(=O)CS(C)(=O)=O)C(F)(F)CC1 C1(C(=O)NCC2(F)CC(CNC(C)=O)C2)CCCC(C)(C)CC1 c1(OC)cc(C(=O)NCC2(NCCO)CC(C)C2)ccc1OC.c1(C)nnnn1C NC(=O)CCC(=O)NC1CCC1NC(c1cnc(-c2ccccc2F)s1)=O c1(C(N2CC(C(C)NC(C3C(C=C(C)C)C3(C)C)=O)C2)=O)cc(C)ncc1C c1(C(=O)Nc2ccc(NCC3CC3)c(O)c2)c[nH]c2ccc([N+](=O)[O-])cc12 CC1(C)OC2CC(C(N3CCCCC3CNC(=O)CC3CCC(=O)N3)=O)CC2O1 CCC(C)(CC)C(=O)N1CCC(C)C(CNC(c2cccc(F)c2Cl)=O)C1 c1(CC(=O)NCC2CC(O)(CNC(C3(CC)CC3)=O)C2)cc(O)nnc1O.C1CC1 C1(C)(CC(=O)NCCC2(OC)CCC2)CCN(C(c2cc(C)co2)=O)C1 c1(N2CCC(N(CCC)C(C3CCCCC3)=O)C2)ncc(Cl)cn1 c1(C(N(CCOCCNC(C(c2ccccc2)C)=O)C)=O)c(O)cc(O)cc1O c1(OC)ccc(C(N2CCC(N(C(=O)C(C)N(C)C)CC3CC3)C2)=O)c(C)n1 Cc1cc(F)c(CC(N2CCC(C)(CNC(c3ccc(O)cn3)=O)C2)=O)cc1F c1(CC)cc(CC(N2CC3CC3(NC(=O)C(N3CCC(O)CC3)C)C2)=O)n(C)n1 C1(C(=O)NC(CNC(CCOCC(C)C)=O)C2CCC2)COCC(C)(C)O1 C(CCCCCF)NC(C1CC2CC1(c1ccc(F)cc1)C2)=O c1(OC)c(C(=O)NC(CNC(c2ccn(C)c2)=O)CC(C)C)sc(Cl)c1Cl N1(C(C2(C)CCCCCC2)=O)CC2CCC1CC2NC(=O)C1=CCCC1 C1(NC(CCCC#C)=O)C(C)CCN(C(c2ccc(-c3ncon3)cc2)=O)C1C N1(CC(=O)NC2C(CC)CN(C(C3CCCCN3C)=O)C2)CCCNS1(=O)=O N1(C(C(CNC(C2C(CCC)CCC2)=O)N(C)C)=O)CCC(O)(CSC)CC1 c1(OC)ccc(C(N2CC(NC(=O)C3=CCSC3)C(C)C2)=O)n2nccc12 Cc1cc(CC(N2CC(CNC(c3n[nH]c(C)c3Cl)=O)CC2C)=O)cc(C)c1 C1(NC(C2(OC)CCSC2)=O)CCCN(C(=O)CN(C2CCSC2)C)CC1 C12C3CCCCN(C13)C2=O.CC(F)CC(=O)NCC12CC(F)(C1)C2 Cc1ccc(-n2cc(C(=O)NCC(CO)NC(c3ccc(O)cn3)=O)nn2)cc1 C(=O)(CC(CC)CCCC)N1CC(CC=C)(NC(C2CCCC(O)C2)=O)C1 c1(C(N2CC(OCCNC(C(CC)CC(C)C)=O)C2)=O)cnc2nccnc2c1 n1(CC(N2CCC(NC(CCCC(N)=O)=O)C23CC3)=O)nc2n(c1=O)CCCC2 c1(C(N2CCCC(C(C)NC(C3CCOC3)=O)C2)=O)ccc2c(c1)OC(C)(C)O2 c1(CC(=O)N(CCN(C(CC(C)c2ccncc2)=O)C)C)ccc(Br)cc1 N1(C(C2CCC(NC(C3CC(C4CC4)C3)=O)C2)=O)CC2(CSC2)C1 c1(C(=O)NCC(C)CNC(C2COC(=O)N2)=O)ccc(OCCF)cn1 N1(C(C2CC(NC(c3c(F)ccc(C)n3)=O)C23CCC3)=O)CC(C2CCCC2)C1 N1(C(C2C(CC)N(C)CC2)=O)CCC2(CCCN(C(=O)Cn3ccnc3C)C2)C1 C1(CC(=O)N(C(C)CCNC(=O)C(C2CCOCC2)F)C)CCCCN1C n1(C(C)C)nnnc1C(C)(CNC(C)=O)NCc1ccc(C(N)=O)o1 CC1=C(C(=O)N2CCC(NC(c3cc(N)c(O)c(F)c3)=O)C2C)CCC(C)(C)C1 c1(C(C(=O)NCC(=C2CN(C(c3scc(C)c3)=O)C2)F)C)cc2ccccc2o1 C(=O)(C(C)(C)CC(=O)NC1CC=C(C(=O)NCC2CCN(C)C2)C1)OC c1(C(C)NC(N(CC#C)C(C)C)=O)nc(C)c(C(=O)OC(C)(C)C)s1 Cc1cc(OC(C)C)ccc1NC(C1(C(=O)O)CC=CC1)=O N1(CC2(c3ccccc3)C(C)(C)C2)CC2(CCC2)C1.C12CC1C(=O)N2 C(=O)(CCC(CC)NC(C1(C)CCCCCC1)=O)N(CC#C)Cc1ccco1 c1(C(N2CC(CNC(C(C(COC)C)C)=O)C2)=O)c(Br)ccc2n[nH]cc12 Cc1cc(=NC2CN(C(c3cccn(O)c3=O)=O)CC2C)[nH]c(Cl)n1 N1(C(CCc2ccc(=N)[nH]c2)=O)CCN(C(=O)C2=CCCCC2)C2CC12 c1(C(=O)NCCN(C(C2C(SC)CCC2)=O)C)cnc2c(ccn2C)c1 c1(C(N2CC(NC(C3(CC#C)CCC3)=O)C(C)C2)=O)cc2ccc(Cl)c(F)c2[nH]1 N1(CC(c2ccc(F)c(Cl)c2)(F)F)CCC(C2CC2(F)F)CC1 C1(C(=O)OC)CC2(CCCCC2)CN1C(C1CC(O)(C(F)F)C1)=O C(=O)(CCS(=O)(=O)N(C)C)NCC1C(NC(CC2C(C)=NOC2=O)=O)C1 CC1CCCC1(C)NC(c1cc(Br)cs1)=O.c12nc(no1)C(C)OC2 N1(C(c2ccc(CC(C)(C)O)s2)=O)CCC(C)(CNC(C2(CF)CC2)=O)C1 N1(C(C(C(C)O)C)=O)CCN(C(=O)CNC(=O)NCC#N)CC1C c1(C(=O)NCCN(C(c2ccc(CC)c(F)c2)=O)C)c(C)cc(C)c(Br)c1C c1(C2CCN(C(c3c(C(=O)O)ncs3)=O)CC2)ccc(F)c(F)c1 C1(NC(C2N(C)CCN(C(c3ccnc(CO)c3)=O)C2)=O)CCc2nncn2C1 C1(C(=O)NC2(C)CC(F)(F)C2)CC(NC(c2cnns2)=O)C12CCC2 C1(OC)CCCCC1CNC(=O)CC(C)(C)NC(c1nc(C)oc1C)=O Cc1ccc(F)cc1C1(CCN(C(C2COC(C3CC3)C2)=O)C2CC2)CC1 Cc1cccn2cc(CC(=O)NCCNC(C3(CF)CC3)=O)nc12 c1(C(N(C(C(N2CCC(C=C)C2)=O)C)C2CC2)=O)ccn2nccc2c1 C1(C(CNC(C(N(C)C)C2CC2)=O)F)CCN(C(C23COC(CF)(C2)C3)=O)CC1 c1(C(N2CC(NC(=O)CCc3cncnc3)C2)=O)ccc(SC(F)(F)F)cc1 c1(C(N(C2C3CN(C(=O)C(C)(C)NS(C)(=O)=O)CC23)C)=O)cc2ccccc2[nH]1 C1(NC(C2COCCN(C(C34C=CC(CC3)C4)=O)C2)=O)(CO)CCC(F)(F)CC1 c1(NC(C2(C)C(C)(C)C2)=O)cccc(CNC(c2cnn(C3COC3)c2)=O)c1 N1(C(c2c(C)sc(O)n2)=O)CC(NC(=O)CN2CC3CC3C2)CC12CCOCC2 C=CC(C)CC(=O)NCC1(C)CCCN1C(c1csc(-c2ncccn2)n1)=O C(=O)(C1=NOC(C(=O)NCCNC(=O)COCCOCCO)C1)C1(C)CCC1 CC(C)C(F)C(=O)NCc1nocc1C(N1CCOCC1C(C)O)=O N1(C(C2CC(=C)C2)=O)CCC2C1CCCN2C(c1cccc([N+](=O)[O-])c1)CC c1(OC(C)C)ccc(N)c(C(=O)NC2CN(C(c3csc(C(F)F)c3)=O)C2)c1 Cn1cc(C(=O)NCCc2ccc(C(F)(F)F)nc2)c2cccnc12 C1(NC(C2C(C)(C)C2)=O)CCN(C(c2ccc(C3CCCO3)[nH]2)=O)CCC1CO C(C)(CCCC(=O)NCC1CC(O)C1(C)C)NC(CC(C)C)=O C1(N(C)C(C2CC3(CC3)C2)=O)CCC(NC(C2CC2C2CCCO2)=O)CC1 c1(C(N2CC(F)(CNC(CN3C(C)CC3)=O)C2)=O)ccc(C(C)(F)F)cn1 CC(C)(C(F)(F)F)OCC(=O)N(CCNC(=O)CCC1CCC(=O)N1)C1CC1 c1(-n2cc(CN3CCC(NC(C(C(C)C)N(C)C)=O)C3)nn2)ncc(Cl)cc1Cl c1(CNC(c2ccc(C)o2)CCOC)cc(C(=O)O)ncc1F CCCCCC(C)CC(=O)NC1(COC)CCN(C(C2CC(CC)C2)=O)CC1 C(=O)(C(C)C1=CCCC1)N(CC(C)CNC(c1nc(Cl)sc1Cl)=O)C C1(NC(C(CC#C)CC#C)=O)CN(C(=O)C(N)=O)Cc2ccnn2C1 c1(C(N(C)CC2CCCN2c2nc3ccccc3s2)=O)ccc2cccnn12 C1(NC(C(N2CCC(O)CC2)C)=O)CC(C2CC(O)C2)C1 c1(C(=O)NC2C(CNC(=O)CCc3ccncn3)C2)ccc(OC(F)F)nc1Cl C(=O)(C1=CCCCC1)NC(C)C=CC(N1CCCC1C1(C2CCC2)CC1)=O C1(NC(c2ccc(COC)s2)=O)CC(NC(=O)CSC)C12CCOCC2 c1(C(=O)NC2CCN(C(C(CC)O)=O)C2)[nH]c(C)c(S(N)(=O)=O)c1C N1(C(CNC(=O)OCC)=O)CCN(C)C(C(=O)NCCC(C)C(F)F)C1 CCC(C)(CNC(c1ccccc1)=O)C(=O)N1CCC(O)CC1CO C12(C(=O)NC3CCC(N(C(Cc4ncc(CC)[nH]4)=O)C)CC3)CC1COC2(C)C C1(C(=O)NCc2cncs2)CC(O)CCN1Cc1cc(I)ccc1Br N1(CC)CC(NC(C2CCC(C)N2C(c2c[nH]nc2C)=O)=O)CCC1=O C1(O)(c2cn(CCCN(C(c3c(C)[nH]c(=N)s3)=O)C3CC3)nn2)CC2CCC1C2 n1(CC)ccc(C(=O)NCCC(=O)NCc2ccoc2C)n1 c1(C(=O)NC(C2CCN(CCNC)CC2)C)cc2cccc(OC)c2o1 c1(OC)cccc(NCC(C)(C)C)c1.c1(N2CC2=O)ccc(F)cc1 N1(C(C2N(C(c3nn(C)c(Cl)c3)=O)CC2)=O)CC(=O)N2CCCC2C1 c1(C(N2CC(OCCNC(C3C(C(=O)OC)C3)=O)C2)=O)cnccc1C(F)F C1(NC(C=CC)=O)CC(C(F)F)(NC(=O)C=Cc2nccs2)C1 N1(C(C(C)OCC)=O)CC(C)(C)CC1CNC(c1ccc(CC(F)(F)F)cc1)=O CC(CCC(C)(C)C)NC(=O)C(CNC(C1CC1(C)C)=O)N(C)C C1(C#N)(C(N(CCNC(COCCC=C)=O)C)=O)CC12CCOCC2 CC1(OCC(=O)NCC2(NC(C3(O)CCOC3)=O)CCC2)CCOCC1 CC(C)C(C(=O)NCCOCCNC(=O)CN1CCCC1C)NS(C)(=O)=O C1(C(N2CCC(OCCNC(=O)C3=NOCC3)C2)=O)CCc2ccnn2C1 CCN=c1[nH]c(C(N2CCC(CNC(c3cnn(CC(C)C)c3)=O)CC2)=O)cs1 C1(CC)CCN(C(=O)CC2CCCC(C)C2)C1CNC(c1sccc1Cl)=O C(=O)(N1CC=CCO1)C1NCCC1.c12nocc1CC(C)(C)n1cc-2nn1 N1(C(C2C(COC)C2)=O)CCN(C(C)=O)CC1C1CC1.C12(CC1)CC(=O)N2 Cc1nc(C)c(C(=O)NC2CCCC(NC(=O)CC(F)(F)F)C2)c(C)n1 c1(C(C)F)ccc(C(=O)NC(C2CCCN2C(c2cc[nH]c2C2CC2)=O)C)cc1 C1(C(N2CC(C)N(C(c3nnsc3C(F)F)=O)CC2)=O)CCc2ncccc2C1 C=C(C)C(C)(C)C(=O)NC(CN(C)C(C1CC1CCC)=O)Cc1ccccc1 C1(NC(C2C3(CC(OCC)C3)C2)=O)CC2CCC(C1)N2C(C12COCC(C1)C2)=O C1(C(N2CCC(n3cnnn3)C2)=O)CSCN1C(c1cc(C(F)F)no1)=O CCC(CNC(=O)C(CC(C)C)NC(=O)C(O)CCSC)CC(C)C CC1(C)CC(NC(C2C3CCC2CC3)=O)CN1C(c1ccc(C#N)cc1)=O c1(C(N2CC(F)(CNC(CS(CC)(=O)=O)=O)C2)=O)nn(C)c2ccc(F)cc12 C#Cc1cc(F)ccc1NC(c1ccc(Cl)o1)=O c1(C(=O)OCc2cnc(=N)[nH]c2)ccc2ocnc2c1 Cc1ncc(C(N2CC(F)(C(=O)NCC(CO)C(C)C)C2)=O)c(=N)[nH]1 C1(C)(C(N(CC(C)(C)NC(C(c2cnn(C)c2)C)=O)C)=O)CC=CCO1 C1(NC(CC2(CC)CCC2)=O)CC(CC(=O)NCc2occc2C)C1(C)C N1(C(C(CCC)C)=O)CCN(C(=O)CN(c2ccc(Cl)cc2)C)CC1CC C(=O)(CC(C)c1cnn(C)c1)NCCN(CCOC)C(C1CC1(C)C)=O Cc1nc(C)c(CC(=O)NC2CCN(C(=O)C(C)(C)c3cnco3)CC2)c(O)n1 Cc1cc(C)c(C(=O)NCCCN(CCCNC(C2CCCO2)=O)C)c(O)c1 c1(C(=O)NC(C)CNC(c2c(Cl)cccc2Cl)=O)ccc2nc[nH]c2n1 CC1(C)OC2(CO)CC1(C(N1CCC(NC(C3(Cl)CC3(F)F)=O)CC1)=O)C2 CC1CN(C(=O)CSCc2ccc(F)cc2)CC1NC(C1COCCOC1)=O C(=O)(NNc1ccc(C(=O)O)c(Cl)c1)NC1(c2cn(C)nc2)CCCO1 c1(-n2cc(CCCCNC(C(CCOC)C)=O)nn2)cccc(Cl)c1OC C1(C(N2CC(C)(C)C2)=O)CN(C(C2CCCCO2)=O)CCC1(C)C C(=O)(CCCCCCS(N)(=O)=O)N1CC(CCNC(C(C)C2CCOC2)=O)C1 c1(SCC(C(=O)N(C(C)C)CCNC(=O)C(C)(O)C2CCC2)C)ccc(F)cc1 Cc1cc(NC(=O)C(C2CCCN(C(C3CCCCO3)=O)C2)(C)C)c(C)s1 S(=O)(=O)(c1cnccc1N(C)Cc1ccc(C)s1)N1C(C(=O)NC)C=CC1 c1(C(=O)NCC23CC2CN(C(c2cc(Br)no2)=O)C3)ccn2cncc2c1 c1(NC(=O)CCCF)cccc(NC(c2coc(C(N)=O)c2)=O)c1 c1(CCCNC(C2(C(F)(F)F)CCC2)=O)cn(CC2CCCC2)nn1 c1(C(N(C)CC2CCN(Cc3ccc(COC)o3)C2)=O)noc2c1COCC2 Cc1ccc(C2CC2C(=O)N(CCNC(C2CC3C=CC2C3)=O)C(C)C)c(F)c1 c1(C(N(CCN(C(=O)CC2CC3CCC2CC3)C)C)=O)ccc2ncccc2n1 N1(S(CC=C)(=O)=O)CC(C(=O)NC(c2cccc(Cl)c2)CC2CC2)C(F)(F)C1 CCCCCC(C)C(=O)N1CCN(C2CCCC2NC(=O)CCCCSC)CC1 C(=O)(C(F)C(=O)NCC(=O)N(C1CN(C(C)=O)C1)C)OCC N1(C(CCSCC)=O)CC(NC(=O)C(c2cc(Cl)ccc2OC)(F)F)C2CC2C1 C#CCC(C(=O)OC)NC(c1nn(Cc2ccccc2)cc1Cl)=O c1(C(N(C2(CNC(=O)CC3CC3)CC2)C)=O)ccoc1C1CC1 Cc1cc(Cl)ccc1CNC(C1NC(=O)CC1C)=O Cc1nc[nH]c(=NCC2CCCC(NC(c3ccc4c(c3)CC(=O)N4)=O)C2)c1Br C(=O)(C(C)CC(F)F)NCCCCC1CCCN(C(CCc2ccc(C)o2)=O)C1 c1(CC)cc(C(=O)NCC(F)CNC(=O)C(CC)c2cccnc2)ncn1 c1(C(=O)NC2C(NC(Cc3ccc(CC)cc3)=O)COCC2)nnc(O)nc1O c1(CNC(N2CCC(N(CCCCOC)C)CC2)=O)cccn(C)c1=O C1(NC(c2cnc(C#N)s2)=O)CCN(C(C2CCCCN2N=O)=O)CC12CCC2 C(=O)(C1=NOC2(CCC2)C1)N1C2CC(NC(C3(NC(C)=O)CCC3)=O)CC1CC2 CCCC(C)CC(=O)NCCC1(O)CCN(C(=O)CCc2cccc(OC)c2)C1 CCC(C)CCCCC(=O)NC1(C2CN(C(=O)C(CCSC)OC)C2)CC1 c1(CSC)ccc2c(c1)CN(C(=O)C=CC(F)(F)F)C2.C1C(=O)N1 C(C)(CC(C)C(F)F)NC(C(C1CN(C(c2ccnc(C)c2C)=O)C1)OC)=O CC1CN(C(=O)C(=O)NCC(F)F)CC1(C)CNC(=O)Cc1ccsn1 n1(C(CC)(C)C)nnnc1C(c1cccs1)NCCCn1ccnc1 C1(C(=O)NCC#C)CN(C(=O)C(CCOC)OC)CC(C)O1 N1(C(c2cnc(OC)nc2)=O)CC2CCC(CNC(=O)C3=C(C)CCOC3)C2C1 Cc1cc(C(N2CC3CC2CC3CNC(=O)C=CC(C)C)=O)c2ncccc2c1 C1(NC(C2N(C(CN3CC(C)(OC)C3)=O)CC2C)=O)COCC(C)(C)C1 CCCCC(CNC(=O)CNC=O)NC(=O)Cc1cnccn1 C1(CNC(c2ccc(Cl)cc2)=O)CC2(CCN(C(=O)C=CC3CC3)CC2)CO1 CCCC(C(=O)OC)C(=O)N1CC(NC(=O)C(F)(F)C2(O)CCC2)C(C)(C)C1 c1(C(=O)NCCN(C(c2cc(OC)ncc2Cl)=O)C)ccc(C)c2ncccc12 N1(C(c2c([N+](=O)[O-])cn(C)n2)=O)CC(N=c2nc[nH]cc2C#N)C(C)(C)C1 C1(NC(C(N2CCC(O)CC2)C)=O)C2CCCN(C(=O)C(F)C(F)(F)F)C2C1(C)C CC12CSCC1CN(C(c1cccc(-n3cc(-c4ccncc4)nn3)c1)=O)C2 c1(C(N(C(C)CNC(=O)CNC(c2cscn2)=O)C)=O)cn(C)c(=O)n1C c1(C(=O)NCCC(=C)CNC(c2ccnnc2C)=O)ccc(C)c2c1CCC2 CC1(C(=O)NCC2(CNC(C3CCCCC3O)=O)CC2)COc2ccccc2O1 N1(C(C2CCCCN2Cc2cccc(F)c2)=O)CCCC2(CCOC2Br)C1 c1(C(=O)NCC2C(NC(CCCCCNC(N)=O)=O)C2)ccc2n[nH]cc2c1 c1(C(N2CC3CCN(S(=O)(=O)CC4CC4)CC3C2)=O)cc(Br)c2ccccc2c1 CC1CN(C(C23CSC(C2)C3)=O)CCC1NC(C1CCN(C2CC2)CC1)=O C(=O)(C(CC=C(Cl)Cl)c1ccccc1)N1CCC(NC(=O)CCC2CC2)C12CC2 C1(CC=C)(NC(C2CCS(=O)(=O)N2)=O)CCCN(C(=O)C(c2ccccn2)O)C1 CC1CN(C(c2[nH]nnc2C2CC2)=O)CC1(C)CNC(c1ccc(F)c(F)c1)=O c1(C(C)C)ccc2cc(C(=O)NC(C3CCCC3O)C)[nH]c2c1 n1(CC(N2CC(NC(C(CC=CC)C)=O)C2)=O)nc(C)c(C=NO)c1C N1(C(CC2CN(C)C2)=O)CC2CC(NC(C3CC4C(C3)C4(F)F)=O)CC1C2 C1(C(C)NC(=O)CCCN2CCCCC2)CCCCN1C(C1CCCC1C)=O Cc1sc(C(=O)NCC2(CO)CCNC2)nc1C(C)C CC1CC(NC(=O)CCC2CCCO2)CN(C(C2(Nc3ccccc3)CC2)=O)C1 C1(C(=O)NCC(CNC(CC=C(C)C)=O)C)CC(c2ccc(F)cc2)=NO1 c1(COC)nc(C(=O)N(C)CCOCCNC(=O)CCCc2cccs2)n[nH]1 C(=O)(CCCCCNC(C1CCCCS1)=O)N1CCC(OCC)C1 C(=O)(CC(C)C(C)C)NC1(CC=C)CN(C(=O)CNS(=O)(=O)C2CC2)C1 C(=O)(C(C)C(F)(F)C(F)F)N1CC(CCC)C(NC(=O)CC(CC)SC)C1 N1(CC(=O)NC(C2CN(C(=O)CN3CCCC3=O)C2)C)CCCCC1C N1(C(c2ccc(CCC)s2)=O)CC(NC(=O)CCCOC(C)C)CC(C)C1 C1(NC(C(C)n2cccn2)=O)CC12CC(NC(=O)COC1CC=CC1)C2 CC(C)CC(C)CC(=O)NCC12CCC(CC1)CN2C(c1cccn1C)=O c1(C(=O)NC2(CF)CCN(C(CC(=O)NC)=O)C2)coc2c1CCCC2 N1(C(CNC(=O)OCC)=O)CCC(C(N2CC(c3ccccc3)C2)=O)(CO)C1 C1(NC(C(C)S)=O)CC2CCC(C1)N2C(=O)Cc1ccc(F)c(F)c1 N1(C(CCOCCCOC)=O)CCOCC1CCNC(C1CC(F)(CO)C1)=O Cc1ccc(NCCC(=O)Nc2cccnc2)c2[nH]ncc12 C1(F)(CNC(=O)C=CBr)CC(NC(=O)CCSc2ccccc2)C1 N1(C(c2cncc(C)c2Cl)=O)CCC2(CCN(C(=O)C=Cc3cscn3)CC2)C1 c1(C(C)=O)cccc(OCC(=O)NCCCCCN(C)C(C2(N(C)C)CC2)=O)c1 C1(F)(CNC(c2nc(C)sc2)=O)CCN(C(=O)CS(C)(=O)=O)C1 c1(C(=O)OCC)cc(-n2cc(C(=O)CN3CCC(C)CC3)nn2)cc(Cl)c1 C1(NC(C(N2CCC(O)CC2)C)=O)CN(C(C2CCNC2=O)=O)C(C)(C)C1 C1(F)(C(=O)NCC(CO)NC(C23C(C(N)=O)(CCC2)C3)=O)CC2(CCC2)C1 c1(C(N(C2CC(NC(C3CC(=O)OC3(C)C)=O)C2)C)=O)ccn2cnnc2c1 c1(N2CC(COC)N(C(c3ccsc3)=O)CC2)ncc2c(Br)cccc2n1 N1(C(Cc2n(C)ncc2Cl)=O)CCC2(NC(c3nccc(C4CC4)n3)=O)CC2C1 c1(CN(C(CCNC(=O)OCC)=O)C)cccc(C(C)(C)CO)c1 C1(O)(C(=O)OCC)CCN(C2CCCC2c2ccc(Cl)cc2)C1 C1(CCNC(C(CC)=CC)=O)CCCN(C(c2cn(CC)cn2)=O)CC1 C(=O)(C1CCCc2scnc21)NC(C1CCN(C(C(CC)SC)=O)CC1)(C)C Cn1cnc2cccc(C(N3CCOC(Cn4cc(CCCCO)nn4)C3)=O)c12 N1(C(C(CC)OC)=O)CC(O)CC1C(=O)NOCCOCCOC c1(C(=O)NC(CNC(c2c(C)csc2)=O)CO)csc2cc(Cl)ccc12 c1(NC(=O)OCC)ccc(NCC(c2cccc(OC)n2)(F)F)cc1C#N c1(CSc2n(-c3c(C)cccc3)nnn2)ccc2c(c1)C(=O)NC2=O c1(COc2ccc(OC)cc2)c(C(=O)O)ccc(Br)c1C.C1CO1 C12(NC(c3n(CC)nnc3)=O)CCC(CNC(C3CC4CC(=O)C3C4)=O)(C1)OC2 C1(OC)CC(C(N2CC(O)(C(C)(C)CNC(C3(CC#N)COC3)=O)C2)=O)C1(C)C CCC(C)CC(C(=O)NCCC1(C)CCOC1)NC(c1cccc(=O)o1)=O N1(C(C2C(N(C(C)=O)CCO)CC=CC2)=O)Cc2ccc(C)nc2C1 O(N(C)C(=O)C(C)CCCC(C)C)CC(=O)OC.C12(CC(O)C1)C(=O)N2 c1(SCC(=O)N(C2CN(C(c3cc4cscc4s3)=O)C2)C)ncnc2[nH]cnc12 c1(OC)cc(CN2CC3CCC2CN3C(=O)CN2C(=O)C=CC2=O)cc(F)c1O C1(CC(=O)N(CC)CC2CCCO2)CC(C)(C)CN1C(C1CC(C(C)C)=NO1)=O C1(NC(c2cc(CC)[nH]n2)=O)CC2CC(NC(c3ccn(C4CC4)n3)=O)CC2C1 Cc1ncc2n1CCC(C(=O)NC1COCCC1NC(=O)Cc1cncs1)C2 C(=O)(C1=NNC(=O)C1)N(CCNC(CCCOC1CCC(C)CC1)=O)C C1(NC(CSC)=O)CC(CNC(c2oc(C(F)(F)F)nc2C)=O)CC1O c1(C(=O)NC2(CNC(C3C=CCCC3)=O)CCOC2)cnccc1Cl C1(CNC(c2nc(C(C)OCC)sc2)=O)CN(C(c2nc(C)c(C)s2)=O)CC1C c1(C(N2CCC(O)(CNC(c3occc3Cl)=O)C2)=O)cccc(F)c1C1CC1 C1(C(=O)NCC(C)CCCO)CCCN(C(c2cn(CCO)nn2)=O)CC1 C1(NC(C2(C)CC=C(C)CC2)=O)CCC2CCN(C(c3cc(Cl)ccn3)=O)C1C2 c1(C(N(CCNC(C2(C)CCOCC2)=O)CC)=O)cc(Br)c2nccn2c1 c1(C(N(CCNC(c2ccc(COC)[nH]2)=O)C)=O)ccn2ccnc2n1 Cc1cc(Cl)cc(C(=O)NCCC(C(C)C)NC(C2CC3CCC2CC3)=O)c1C C(C(C(=O)N(C1CCCOC1)C)C(C)C)NC(C(COC)OC)=O c1(CC)ccc(C(C)=CC(=O)NC2CC(O)CN(C(c3ocnc3C)=O)C2)cc1 N1(CCCC)CC2(CCC2)C1C1CCN(C(c2ccn(C(C)C)n2)=O)CC1 C1(NC(c2ccc(OC)nn2)=O)COC2(CCN(C(=O)Cc3cnc(C)[nH]3)C2)C1 c1(C(F)F)cccc(C23CC2CCN3)n1 Cc1ccc(-n2cc(C3CCN(C(=O)CCF)C(C)C3)nn2)cc1F C(=O)(C1CCCn2cnnc21)N1CCN(C(=O)C=CC2CC2)CC(CO)C1 C1(=CC(=O)NC(C)C(CO)NC(=O)C(=O)NCC(F)F)CN2CCC1CC2 C12(NC(C3(CC=C)CCCN3C(=O)CCN(C)C)=O)CCCN(CC1)C2 Cc1nc(C)c(-c2nc(CCC(C)C)nn2-c2cccc(C(C)C)c2)o1 c1(C(=O)NCC2(NC(C(CCC)CC)=O)CCC2)cc2c(cc1Cl)OCO2 C(=O)(CC(CC)C(C)C)NC(CC(=O)N(CCC)CCN(C)C)C(F)F Cc1nc(Cl)ncc1NC(=O)CC12CCC1CN(C(=O)C1=C(Cl)CCC1)C2 c1(CC(C)C(=O)N2CCC2CNC(c2ccc(Cl)nc2O)=O)ccc(C#N)cc1 c1(OCCN(C(C(=O)NC(CNC(COC)=O)C)CO)C)ccc(Cl)cc1 CN1CCC(NC(=O)Nc2cccc(OC3CCCCC3)c2)C1=O c1(C(=O)NCC2(CO)CCN(C(c3nc(CC)oc3)=O)C2)ccc(N)c(C)c1C C1(NC(C(c2scc(C)n2)C)=O)(CNC(C2C(C)C2C)=O)CCOCC1 c1(C(N2CCC(OCCNC(=O)C=C(Cl)Cl)C2)=O)nccc(C(F)(F)F)n1 C1(NC(=O)COCCc2ccc(Cl)s2)CCCCN(C(=O)C2=CCOCC2)C1 c1(OCCNC(CN(C(=O)OC)C)=O)cn2c3c(cc(F)cc3c1=O)CCC2C CC1(CC(N2CC(O)(CNC(=O)CC3CC4(CC4)C3)C2)=O)CCCCC1 C12(NC(C(=O)NCC)=O)CCCCCC1N(C(c1csc(C(C)(C)C)c1)=O)CC2 c1(C(N2CCC(N(C(C3(CC#C)CC3)=O)C)CC2)=O)ccc(Br)nc1N n1(C(C)(C)C)cccc(C(N2CC3CC(NC(C4CC(F)C4)=O)C3C2)=O)c1=O C1(C(=O)NC2CCC(O)C2)C2CN(C(C3CN4CCC3C4)=O)CC12 c1(C(C)NC(=O)CNc2sccc2C#N)ccc(F)cc1Br C1(NC(c2csc(-c3ccsc3)n2)=O)C=CCN(C(C2CC2F)=O)C1 N1(C(C(C)Cc2cnc[nH]2)=O)CCC(C)C1CNC(=O)C=CC1CCCC1 c1(OC)cc(=NC(=O)CC2CC(NC(=O)C(C)(C)CC#N)C2(C)C)[nH]n1C C1(CC(C)C)COCC1NCc1noc(C(F)F)n1 N1(C(C(CC)(C)CC)=O)CCCC(C2CC2NC(=O)CCc2cccs2)C1 C1(C(C)C(=O)N(CC(=O)O)CC2CC2)CCCCCC1 C(=O)(C1CNS(=O)(=O)c2ccccc21)NC1(C)CCOC12CC2(F)F C(=O)(C1=NN(C2CC2)C(=O)CC1)N(C1CCC(NC(=O)C=CC(F)(F)F)CC1)C C(=O)(C(O)CC(C)(C)C)NC(CCCC)CNC(=O)COc1ccc(Cl)c(F)c1 N1(C(C(CCCC)NC(C2CC(C3CC3)C2)=O)=O)CCC2(CNC(=O)N2)C1 c1(-c2cccc(NC(C(=O)NC3CC(C)(CC)C3)=O)c2)cn2ccsc2n1 C(=O)(C1CCCc2c1ncn2C)N1C(CN(C(c2n(CC)cnn2)=O)C)CCC1 C(=O)(C(C)(C)CC(=O)NC1CCN(C(=O)Nc2cccc(F)c2)CC1O)OC C1(CC)CC(O)CN1C(=O)CC(C)CNC(C1CC(OC)C1)=O c1(NC(C2CC(F)(F)CN2Cc2ccccn2)=O)cc(F)c(F)c(F)c1 C1(CNC(C(C)c2ccsn2)=O)CN(C(=O)CCc2cn[nH]c2)CC1C C1(NC(CC2(C=C)CN(C(=O)CCCC#N)C2)=O)CCOC(C)(CC)C1 N1(C(C=Cc2ccc(C)o2)=O)CCOCC(C(=O)NCc2cscc2C)C1 c1(C(=O)NCCC(C)NC(C2CC23CCC3)=O)csc2nccn12 Cc1c(C(=O)NCC(C2(O)CCN(C(C3(CN(C)C)CC3)=O)C2)C)nnn1C c1(C(=O)NCC2CN(C(C3ON=C(C)C3)=O)CC23CC3)cc(C#N)cc(C)n1 C#CCCCCCC(C(=O)O)NC(c1cc(CN)ccc1O)=O CCC(CC(=O)N1CC(CNC(c2cccc(OC(F)F)n2)=O)C(C)C1)C1CC1 OC1C(O)C2CC(NC(c3cccc(SCCO)c3)=O)C1O2 C=CCCCC(C(=O)NCc1ccc(C#N)cc1)NC(C1CC2OC1C1CC21)=O CC(CC(C)(C)C)C(=O)N1CCCC(C(C)NC(c2ccc(N)cc2O)=O)C1 C(=O)(C(C)CC(N)=O)N1CCC(CN(C(CCNC(=O)OC)=O)C2CC2)CC1 c1(C(=O)OC)ccc(C(=O)NNC(=O)C2CC2F)cc1 N(C1CCCc2occc21)C(C=C(C)CNC(=O)CC1CCC1C)=O C(=O)(C1=CCC(C)CC1)NC(c1cnn(C)c1)C(=O)NC(CC=C)(C)C(F)F c1(C(=O)NCC2C(CNC(CCC3CC(C)C3)=O)C2)ccnc(C(N)=O)c1 C(=O)(C(F)(CNC(=O)Cc1ccon1)C(C)C)NC1CCCC(C=C)C1 C(CO)(C(=O)NCCC1CC(C(=O)NCCCOCCO)C1)NC(N)=O c1(OC)cc(O)ccc1NC(C1CC(O)CN1C(C1CCCS1)=O)=O C1(C(=O)NC)CCCN(C(c2cnc(C)s2)C(=O)NCCCOC)C1 c1(C(C)(C)C)ccc(CC(=O)NC2CC(CCNC(=O)CCC(F)F)C2)cc1 c1(C(N(CCCNC(c2cnn(C(F)F)c2)=O)C)=O)cccc(-n2ccnc2)c1 c1(CNC(c2n(CCOCC)nnn2)c2sncc2C)cc(C)cnc1Br Nc1nccnc1C(=O)NCC1CCC(CNC(=O)COCC2CCCC2)CC1 C1(C(=O)NCCN(C(=O)C(C)S(N)(=O)=O)CCOC)Cc2nc(C)cn2C1 c1(NC2C(C)CN(C(=O)C3=CCCO3)CC2)ncc2ccnc-2[nH]1 CC(C(=O)N1CC(N2CCN(C(c3sccc3Cl)=O)CC2)C1)C(C)n1cccn1 C1(NC(c2c(C)nc(C)o2)=O)CN(C(=O)Cc2cncnc2)CC12CCC2 CCCC(C(=O)NCC(O)CNC(=O)C=CCN1CCCCC1)NC(C)=O c1(C(N2C(CC(=O)NCc3ncco3)CC(F)C2)=O)cccc(F)c1F CC1CCC(C(=O)NC2(C)CCSC2)CN1C(=O)CCC1(C#N)CCC1 c1(OCC(=O)NC2CC(C(=O)NC(CNC(C)=O)C)C2)cccnc1 c1(OCC(=O)NC2(CCCNC(CC(C=C)C)=O)CC2)cc(F)cc(F)c1 Cc1cnc(C(=O)N(C2(C(N3CC4C(C)C4C3)=O)CCC2)C2CC2)c(C)c1 CCCCCCC(C)C(=O)N1CCOCC1CNC(=O)Cn1nnc(=O)[nH]1 Cc1oc(C(=O)NC(C2CCN(C(c3coc(N(C)C)n3)=O)C2)C)cc1Br C1(CNC(C(C)n2cccn2)=O)CN(C(C2(C3CCC3)CC2)=O)CCCO1 c1(C(=O)NCCC2CN(C(C(COC)N(C)C)=O)C2)cccc(C)c1Cl c1(C(N2CCC(O)(C(C)NC(C3CCC(F)(F)C3)=O)C2)=O)cccc2oncc12 N1(C(C(C=C)OC)=O)CCOCC(COC(=O)COC(F)F)C1 C1(NC(N(C2CCCN(C)C2)C)=O)CCC12CCC1(CC2)OCCO1 N1(CC)CC(C(=O)NCCCNC(=O)CN2CCN(S(C)(=O)=O)CC2)CC1=O C1(C(=O)NCC(CC)(C)NC(=O)Cc2cnn(C)c2C)CC2(CCOCC2)CO1 N1(C(c2n(CC#C)ccc2)=O)CC(CC(=O)N(CC(C)OC)CC)CC1(C)C c1(NC(CC2CN(C(COCC(=O)OC)=O)C2)=O)ccc(C(F)(F)F)nc1C c1(C(=O)NCc2cn(C3CN(C(C(C)CN(C)C)=O)C3)nn2)ncc(Br)cc1O C1(S(C)(=O)=O)(C(N2CC(CNC(C3(C(C)C)CCC3)=O)OCC2)=O)CCC1 C1(CCNC(CC2(OC)CN(C(c3cccc(=O)o3)=O)C2)=O)CCC(C)(C)C1 Cc1cc(CCC(=O)N(C)CC2(CNC(C3C=CCCC3)=O)CC2)n(C)n1 c1(-c2cn(CC3(CC4CC4)CCCC3)nn2)ccccc1F.N12CCCC1NC2=O c1(OC)ccc2[nH]c(C)c(CNCC34CCC3CCN4C(=O)OC(C)(C)C)c2c1 CC1Oc2c(C(=O)NCC3CCN(C(C45CC4C5)=O)C3(C)C)cccc2NC1=O C1(CN(C(CSC)=O)C)CN(C(=O)CCc2cnccn2)CCO1 c1(C(=O)NCC(C)N(C(C2CC(C)(C)CO2)=O)CC)nsc2ccccc12 C(=O)(CS(=O)C(F)(F)F)NCC(CC=C)NC(c1ccc2nccn2c1)=O N1(C(C=COCC)=O)CCC2(CC1)CC(C(=O)NCC1CCCO1)CO2 Cc1nc(=N)[nH]cc1C(N1CCC2(CC2NC(C2CC(O)C2)=O)C1)=O C1(NC(C(C)Oc2ccc(OC)cc2)=O)CN(C(c2ccc[nH]2)=O)CC2(CC2)C1 CC(C)CC(O)CNC(=O)C(CCOCCO)NC(C1OC2CCC1C2)=O N1(C(CN(CCC)C(C2CCCC2C)=O)=O)CCCC(C(=O)OC)C1 c1(C(=O)NC2CCN(C(=O)CCN3CCOCC3)C2)cccc(-c2nccs2)c1 N1(C(C2C(C)(C)CCCO2)=O)CCOC2CN(C(=O)C(F)CC3CCOC3)CC12 C1(C(N2CC3OCC(CNC(=O)OC(C)(C)C)C3C2)=O)CC2CC(=O)CC(C1)C2 C12(C(=O)NCC(C)F)CCC(CN(C(=O)CC3(C)CCOCC3)C1)C2 CCCCCCC(F)C(=O)NC1CC(=O)N(C2CN(C(c3cnccn3)=O)C2)C1 CCCCC(O)CC(=O)NC1(CF)CCN(C(=O)C=CC(N2CCOCC2)=O)C1 C1(C(N2CC(C)(CNC(=O)Cc3cnsc3)OCC2)=O)CCn2cncc2C1 c1(N2CCC(C(=O)OCC)C2)nnc(-c2ccccn2)n1Cc1cccnc1 C(C)(CNC(=O)C=Cc1ccncn1)(CC(C)C)NC(C(CSC)OC)=O C(=O)(C1=CCCSC1)N(C1CCN(C(CC2CCC(=O)CC2)=O)CC1)CC1CC1 C1(S(=O)(=O)CC)(C(=O)OC(c2onc(CC)n2)C)CC1 c1(CC)ccc(C(=O)NCC2(C)CN(C(=O)CC3=CCCC3)CC2C)c(N)c1 CCCC(O)(CCC)CC(=O)NCCCOCCNC(=O)C(CC)NC(=O)OC CCCCC(F)C(=O)N1CCCC(NC(=O)Cc2sc(C)nc2C)C1 N1(C(CCCC#C)=O)CC2CN(C(=O)C(F)CC)CC12 c1(C(=O)NCC2(F)CC(NC(C3(OC)CCOC3)=O)C2)ccncc1O C12(Cn3cc(CN(C)C4CC4)nn3)CC1CN(C(=O)CCC(=O)c1ccccn1)C2 C1(=O)CC(C(C)OC)N1.C1(CC)(CO)CCCN1C(=O)CCOCCCN(C)C CP(C)(=O)C1CCCCN(C(=NCCF)NCC2CC(S(C)(=O)=O)C2)C1 N1(CC(=O)N(CCC(C(C)C)NC(=O)CC2CC23CC3)C)C(=O)CN(C)C1=O C1(NC(c2cc(OCC)no2)=O)CC2CC1CN(C(=O)Cc1ccns1)C2 Cc1c[nH]nc1C(=O)NCC1CC1CNC(=O)CC1(C)CC1(Cl)Cl CS(=O)C1CN(C(=O)C(CC2CCOCC2)NC(=O)CC2CCCC(=O)C2)C1 C(=O)(CC1=CCOCC1)NCC(C(=O)N(CCOC)C)(C)C C12(C(N3CCN(CCNC(=O)Cn4cc(Cl)cn4)CC3)=O)CCCN1CC(O)C2 c1(C(=O)NCC2(NC(C3CN(C)C(=O)N3)=O)CC2)ccc(S(C)(=O)=O)o1 C1(C(N2CCC(C)(NC(c3ccc(NC)cn3)=O)CC2)=O)CCC12CCOCC2 c1(NC(C(CC)C)=O)cscc1C1=CC(=O)CCC1 Cc1cccc(C)c1C(=O)N(C(C)C(N1CC2CC2C2CC12)=O)C1CC1 CCC(C)C(CO)CN=c1ccnc(NC2CCN(C(=O)N(C)C)CC2)[nH]1 C(C)(C(=O)NOC(CC(C)C)C(=O)Nc1ccc(O)cc1OC)=C(C)C CCCC(C(=O)NC12CC(NC(c3ncc(Br)cn3)=O)(C1)C2)OCC c1(C(=O)NC(C2CCN(C(c3n[nH]cc3[N+](=O)[O-])=O)C2)C)ccc(Cl)c(Cl)c1 c1(-c2ccc(C(=O)NCCN(CC(F)F)C)s2)cccc(Cl)c1 n1(CC)cc(CC(=O)NCCC2(NC(c3c[nH]nc3C)=O)CC2)cn1 C(=O)(C(C)C(C)(C)C)NC(CNC(CCCc1onc(CCC)n1)=O)CCOC C1(NC(c2ccc(C)o2)=O)CCN(C(c2cccc(C(C)C)c2F)=O)CC1C c1(CCC(=O)NC2CC(NC(C3CC(=O)C3)=O)C2)ccc2c(c1)OCO2 C1(CC(=O)NCC(C)(C)OCC(=O)N(CC(C)OC)C(C)C)CC(F)(F)C1 Cc1cc(Cl)ccc1OCCCC(=O)N(C1CCN(C(=O)C=CCF)C1)C N1(C(C)=O)CCC(C)(C(=O)NCCN(C(c2cc(N)ccc2C)=O)C2CC2)CC1 c1(C(N(CC(C)NC(COC(CC)CC)=O)C)=O)c(C)noc1N N1(C(C(=O)NCc2cccs2)c2ccon2)CCC(S(=O)(=O)C(F)F)C1 c1(C(=O)NC2CCN(C(C(F)OC)=O)C2(C)C)cnc2[nH]cncc1-2 c1(C(C)C)n[nH]c2nccc(NC(c3ccc4nc(O)oc4c3)=O)c12 C(=O)(CCc1ccon1)NCCN(C(=O)CCC1CC1(F)F)CC(C)O N1(C(Cc2cc(C)[nH]n2)=O)CCCCC1CCCNC(=O)C(c1ccnn1C)C c1(C(=O)NC2CN(C(c3c(C)cc(C)o3)=O)CC2F)scc2c1OCCO2 N1(C(c2c(C(C)C)onc2)=O)CC2CC(NC(=O)CC3=CCCCC3)C(C2)C1 C(CC(C)(C)C(=O)NC(c1cn(C)nn1)CNC(=O)C(C)C(F)F)OC CC#CCCC(=O)N1CC=CC(NC(=O)Cc2ccc(SCC)cc2)C1 c1(Cn2c(Cc3cccnc3)nc(-c3cn(C)nc3)n2)cccc2ncccc12 C(=O)(C(O)C(C)(C)C)N(CCC(=O)Nc1ccc(SC)cn1)CC=C Cc1cccc(C(=O)NCC2CCCC2C(=O)NC2(CC(C)C)CC2)c1 C1(C(=O)NC(CC2CC2)CO)(NC(=O)CSc2cn[nH]c2)CC(F)C1 C1(C(=O)OCCOC(=O)Nc2ccccc2)CCCC(C(=O)NC2CC2)CC1 Cc1cc(C)c(C(=O)NC(C)(C)C(C)NC(c2cc(Cl)ccc2F)=O)cc1N CC(C(F)C(=O)NCCN(C(=O)CCC(=O)c1ccncc1)C1CC1)C(F)(F)F c1(CSCCNC(C(=O)NC(c2nc(C)[nH]n2)C(C)C)=O)ccc(O)cc1 C(CCN=c1nc2c(ncn2C)c(NC2CCC3CCCCC23)[nH]1)OC N1(C(CC)=O)CC(C(=O)NCc2ccccc2OC)CCC1C C(C(C)C(=O)OC)(c1nnnn1C(C)(C)C)NCCC c1(CC)cc(N)c(C(=O)NC2CC(NC(=O)C(c3ccccc3)O)C2)cc1F N1(C(C=Cc2ccn(C)c2)=O)CCC2(CCCC2NC(c2cc[nH]n2)=O)C1 c1(C(N2C(C(N(C)Cc3nnc(C)o3)=O)CC=CC2)=O)c[nH]c2nccc-2c1 c1(C(N2CCC(N(C(C(C)OCC=C)=O)CCC)C2)=O)sc(Br)nc1C C(C(COC)C(=O)NCCc1ocnc1CNC(C1CCC(F)CC1)=O)OC N1(C(C(C)CNC(c2cnn3cccc3c2)=O)=O)CC2(CCC(=O)NC2)C1 N1(C(C(=O)NC(CC)C)CCC2CCOCC2)CCn2c(C)nnc2C1C N1(C(C=CC)=O)CCCC(N(CCO)C(c2cc(C)cs2)=O)C1 C(=O)(C1=CC2CCCC12)NCC12N(C(c3c(C(=O)OC)nccc3)=O)CC(C1)C2 N1(CCC2OCC(C)(C)C2)CC(=O)N(CCC2CCC2(F)F)C1=O C1(C(N2CCC(CN(C)C(C3CCSC3)=O)CC2)=O)CNC(=O)CC1(C)C CC1(C)OCc2cc(C(N3CCC(O)(CCNC(=O)CSC4CC4)C3)=O)ccc21 C1(CC(=O)NCCN(C(c2ccc(=N)[nH]n2)=O)CC)NC(=O)CNC1=O C1(C(N(CCC(C)NC(CS(=O)(=O)NC)=O)C)=O)Cc2nncn2C1 c1(C(N2CC=CC(NC(C(COC)(F)F)=O)C2)=O)ccc(F)cc1OC N1(C(C2CCN(C(CC(C)C)=O)CC2O)=O)CCC2(CCCCC2)CC1 CC(F)(F)C(C)(C)C(=O)NCCCNC(=O)CC1CCC2(CC1)COC2 C1(C)(CC)C=C(C(=O)NC(C)(CNC(C2(c3cccnc3)CC2)=O)CO)C1 N1(C(C(CC(CC)CC)F)=O)C2CCCC1CN(C(=O)CCCCC1CC1)CC2 c1(C(=O)NCCCC(C)NC(C2CC2Br)=O)cc(C(F)F)n(C)n1 CC(F)(F)CCC(=O)NC1CC12CC(NC(=O)CCc1cnc(C3CC3)o1)C2 N1(C(c2c(CC)occ2)=O)CC2CC(NC(c3nc4ncccn4n3)=O)CC1C2 C1(CNC(CCCOCC=C)=O)CCN(c2nnc(-c3ccon3)s2)CC1C c1(CNC(CCC=C)c2nnnn2C2CCCCC2)cnc2sc(Br)cn12 c1(C(=O)NC2CCN(C(C3CCCC(C4CC4)O3)=O)C2)cc(Cl)ccc1F c1(C(=O)NCC(C)NC(c2c(C)ocn2)=O)cccc(F)c1C#N C1(NC(C(CC(C)C)NC(C(C)=CCC)=O)=O)CC2(COCCO2)C1 c1(SC)cccnc1C(=O)NCc1ncccc1C(=O)NN1CC2CC2C1 C1(NC(CSCC=C)=O)CC2CCC1C1CN(C(=O)C(C)C(C)C)CC21 Nc1cnccc1C(=O)NCC1(CNC(=O)C=CC(F)(F)F)CCCCC1 N1(C(CC(COC)OC)=O)CCCCC(CNC(C2(n3cccn3)CC2)=O)C1 c1(C(N2C(CNC(C3CC3C(F)F)=O)CCCC2)=O)cc2c(=O)[nH]ccn2n1 C#CC1(C(=O)NCC2CCCCO2)CCN(C(c2n[nH]c(O)n2)=O)CC1 c1(C(=O)NCC2(COC)CN(C(=O)C(C)CC(C)C)C2)nccc(Cl)c1C Cc1c(C(=O)NCC(CNC(c2cnnn2C)=O)C(F)(F)F)nn2c1CCCC2 N1(C(c2cnc(NCC)s2)=O)CCOCC(NC(=O)CCc2cccc(F)c2)C1 c1(-c2ccc(C(=O)OCCSCCCCC)o2)ccc(COC)cc1 C(=O)(C(C)(O)C(C)C)NCN(CCC)C(C1SCCS1)=O N1(C(=O)CCOCC2CC2)CCOC2(CCCN(C(c3cc(CO)[nH]n3)=O)C2)C1 c1(C(=O)NCC(CC=C)NC(C2CCN2S(C)(=O)=O)=O)cc(C(C)C)[nH]c1CC c1(OC)ncc(C(=O)NC2CC2C(=O)Nc2cnn(CC(F)(F)F)c2)cn1 c1([N+](N2CCOC(O)C2)(C(c2csc(C=O)n2)=O)[O-])ncc(Cl)cc1Cl c1(-c2c(C(N3C(C(N)=O)CCCC3)=O)nccc2)ccc2ncsc2c1 C1(=CC(=O)NCC2CCN(C(C3CCO3)=O)C2)CCOc2ccccc21 C1(C(N(C2CCN(Cc3ncc(C)s3)C2)CCC)=O)CCc2cnc(C)n2C1 C(C(C)(Cn1cccn1)NC(C12CSC(C1)C2)=O)NC(CC1(C)CC1)=O CN1C(=O)C(OC(C2(COCc3ccccc3)CC=CC2)=O)Cc2ccccc21 C1(N(C(c2ccnc(Cl)c2)=O)CC)CCCN(C(C2CC(N(C)C)C2)=O)CC1 c1(C(=O)NCCN(C(COCCCN(C)C)=O)CCC#N)cc2scnc2[nH]1 C1(NC(C2C(C)C2C)=O)CCN(C(=O)Cc2csc(-c3ccccc3)n2)CC1O C(C(C)(C(C)C)NC(=O)Cn1cccn1)NC(C1(OC)CCC1)=O c1(C(=O)NCCC(C)NC(=O)CCC2CCCCC2)ccnc(Cl)c1 c1(C(N2C(CN(C)C(C3(CO)CCCO3)=O)CCCC2)=O)ncc(Cl)cc1Cl c1(CNC(=O)NC(CC)C(N)=O)ccc(-n2cccc2)cc1 C1(CNC(=O)CSc2cccc(F)c2)CC2CCC1N2C(C1(F)CCOCC1)=O CC(C(=O)N(CCNC(=O)C=CSCc1ccco1)CCOCCO)C(C)(C)C Cc1cc(NC(=O)CCCCCN(C)C(c2ncc(F)cc2N)=O)cc(O)c1 c1(C(=O)NC2CN(C(C3CC(O)C3)=O)CC2CC2CC2)cc(O)ncc1Br N1(C(c2ccc(F)c(Cl)c2)=O)CCCN(C(C2CCC=CCCC2)=O)C(CO)C1 c1(C(=O)NCC2(F)CN(C(=O)COC3CC(F)(F)C3)C2)cc2n(c1)CCCC2 c1(NC(CCN(CC(F)F)C(C)=O)=O)cnn(C)c1I Nc1c(C(N2CCCC2CCNC(C2CC2CF)=O)=O)cc(Cl)cc1Cl C1(NC(C(C=C)O)=O)CCN(C(c2snnc2C)=O)CC(C)(C)C1 CN1CC(CNC(C2C(CNC(C3(F)CCCCC3)=O)C2(C)C)=O)CC1=O c1(OC)ccc(OC)c(C(=O)NC(C)CNC(=O)C(c2ccc(O)cc2)(C)C)c1 CCC(O)C(C)(C)C(=O)N(CC(C)(C)CNC(=O)Cc1c(C)nc(O)nc1C)C CC(CC(C)(C)C)C(=O)NCC1CN(C(c2cc(C3CCC3)no2)=O)CC1(C)C N1(CC(=O)NC2(CN(C)C(C34CC(F)C3C4)=O)CC2)C(=O)NC(C)(C)C1=O C1(N(C(C=CC=CCC)=O)C)CN(C(=O)C=Cc2cccc(CO)c2)CC12CC2 N1(C(c2c(C)nc(CC)o2)=O)CC(F)(F)CC1CCNC(C1(CO)CCOC1)=O C1(C(=O)NCC(C(C)C)NC(=O)CCc2ccccc2)CCCCN1C(C)C C(CCCS(C)=O)OC(=O)NC1(C(=O)NC(C)(C)C)CC(OC)C1 CC1CC(=O)NCC1C(=O)NCC(C)(C)CN(C(=O)CCC1CC(F)(F)C1)C N1(C(C(C)(C2CCOCC2)OC)=O)CCOC(CCNC(=O)CC2CCC2)C1 C1(CNC(COC(C)C)=O)CCC(CNC(C23CCC2C3)=O)CC1 CC1C(NC(=O)CC(C2CC2)C2CC2)CCCN1C(=O)CCc1ccccc1 C(=O)(C(C)(C)C(C)NC(=O)C=CC(C)C)NCC(CC)(O)CC C1(CSc2ccn(C)n2)CCC2(CN(C(=O)C(F)CC3CCC3)C2)O1.C1C(=O)N1 c1(C(=O)NC(C=CC(=O)NC(C)C)C)cccc(COC2CCC2)c1 C12(C(=O)NC(CCCC)CCC)CCN(C(c3cc(C)n(C)c3C)=O)CCC1C2 CCCCCCC(CC)NC(C12C(NC(C3CCCC(=O)C3)=O)C3CC1C2C3)=O CC1CCCCCC1NC(C1CCC(CNC(c2ccc(CO)cn2)=O)O1)=O C1(NC(C2CCN(C(C34CCCN(CC3)C4)=O)C2)=O)(CO)CCCCCC1 c1(CC)cc(C(=O)N2CC(n3cc(-c4cccc(CO)c4)nn3)CO2)c(C)nn1 C(c1cncc(O)c1)=CC(=O)NC1CCC(NC(c2n[nH]c3c2CCC3)=O)C1 N1(C(C2N(C(CCCN(C(C)=O)C)=O)CC2)=O)CCCC1(C)CC(C)C c1(C(N2CCC(C3CC3)(CNC(C(CC)SC)=O)C2)=O)cc2ccc(F)cc2o1 N1(C(C(CNC(c2cccc3c2CCC3)=O)O)=O)CCC2(C=CCO2)C1 N1(C(CC(C)C2CCCC2)=O)CCCC(O)(CNC(C2CCC3(CCC3)O2)=O)C1 C1(N(C(=O)NCc2ccc(Cl)cn2)Cc2cccc(F)c2)CCNC2(CC2)C1 C1(C(N(CCCNC(CCCC#C)=O)C(C)C)=O)CC2CCC(C1)N2C C(=O)(CCC(=O)NCC(C)(O)CNC(C1(c2c(Cl)cnn2C)CC1)=O)NCCC n1(CC)nc(C(=O)NCC(CC(C)C)NC(c2n[nH]cc2C)=O)c(C)n1 C(=O)(CCC(F)(F)CN=[N+]=[N-])N(C1CCN(c2ccc([N+](=O)[O-])c(CO)c2)C1)C CC(C)(CC#N)C(=O)NCC1(F)CCC(NC(=O)CCc2ccc(F)cc2)C1 Cc1ccc(C(=O)NC(C)CCNC(=O)C2=CCSC2)cc1S(N)(=O)=O Cc1cc(=NC(=O)C2CCCCN(C(c3cc(CO)on3)=O)C2)[nH]n1C1CC1 c1(C(N(CC(C)N(C(c2ccnc(C)c2C)=O)C)C)=O)cn2c(n1)CCCC2C C(c1ccc(-n2ccnc2)cc1)=CC(=O)NC(C1N(C(CC)=O)CCC1)C C(CC(=O)NCCCn1ccnc1C)(CC(C)C)NC(c1c(C)cc(N)cn1)=O c1(C(=O)NC(CC)(CNC(C2CC2C2CCCO2)=O)CC)cnc(O)c(Cl)c1 C(=O)(CCNC(=O)NCC1CCCO1)C1(C(C)NCC2CSC2)CC1 CC1CC=C(C(=O)NCC#CCNC(c2cc(C3CCCCC3)n(C)n2)=O)CC1 c1(C(C(N2CC(N(C(C3(CC#C)CCCCO3)=O)C)C2)=O)C)cc(F)cc(F)c1 C1(C(N(C(C)CNC(=O)C(COC)OCCO)CC)=O)CCC(C(F)(F)F)CC1 C1(C(C)NCc2scc(CC(=O)N(C3CN(CC)C(=O)C3)C)c2)CC(C2CC2)=NO1 c1(OCCN(C)C)ccc(CNC(=O)Nc2ccc(C(F)(F)F)nc2N)cc1Cl N1(C(Cc2c(C)cccn2)=O)CC2(NC(=O)C3=CCCS3)CCCC2(F)C1 C(=O)(CC(C)(C)O)NCC(C1CC1)NC(CCCOC(CCC)=O)=O Cc1cc(C(=O)NC(Cc2ccoc2)C(=O)NCC(C)(O)CCO)nc(C)n1 n1(CC(=O)N(C2CCN(C(C3(C#N)CC(C)C3)=O)CC2)CC#C)ncccc1=O C1(CC=C)(NC(C2CCC3(CC3)C2)=O)CCN(C(C2CC(CC)=NO2)=O)CC1 C1(C)(NC(c2c(C)nn(C)c2)=O)CCCN(C(=O)C(n2cc(Br)cn2)C)C1 C1(NC(c2n[nH]cc2Cl)=O)CN(C(=O)CCCOc2ccccc2)CC1O c1(CN2CCC(NC(c3cc(C)nnc3)=O)C(O)C2)cc2ccccc2nc1O N1(C(C(CC)NC=O)=O)CCC2(CC(C(=O)NCCOCCOCCO)C2)C1 N#Cc1csc(C(=O)NC2CCCC2NC(=O)C=Cc2ncco2)c1 N1(C(C2C(C(=O)OC)C2)=O)CCC(NC(=O)C2=CC(C)(C)C2)CC1C CC(=O)CC(C)(C)C(=O)NCC1CCC(C(=O)N(C)OC)C1 Cc1cc(C(N2CCN(C(=O)Cc3conc3C)C(CCO)C2)=O)nnc1C C[S+](C)CCC(O)C(=O)NC(C)(C)CCCNC(C1C=CCC1)=O C1(C(N(C2CN(C(=O)C(=O)NCC(F)(F)F)C2)CC)=O)CCC(F)CC1 C1(CNC(COC)=O)CN(C(c2c(C)ncn2O)=O)CC12CCC2 c1(C(N2CC(C)C(CCNC(C3(Cl)CCC3)=O)C2)=O)cc2sccc2[nH]1 C=CC(C)(O)CC(=O)N1CCCCCC1C(N1CCN(CC(C)C)CC1)=O c12cc(no1)O2.C12CC(C1)C(=O)NCC(=O)NCC2.CC(C)(C)CCSC.C1CO1 N1(C(C(C)=CCC)=O)CC(O)(C(F)C(=O)NCCC2(C)CCOC2)C1 C1(C)(C(N(CCN(C)Cc2cn(CCC(=O)OCC)nn2)C)=O)COC(=O)N1 c1(C(=O)NC(c2cn(C3CC3)nn2)(C)C)ccc(-c2cccs2)nc1O c1(CNC(CC2C(C)CCCC2)=O)nn(C)c2c1CN(C(C1C=CCC1)=O)CC2 C(=O)(CCCCN(C(=O)C(C)(C)c1ccsc1)C)NCC1C(C)CC1 c1(C(CN(CC(C)C)C(=O)C2CC2)C)ccccc1Cl c1(C(=O)NCC2CCC(NC(C3C(C)OC(C)C3)=O)CC2)cnc2[nH]ncc2c1 c1(CC(C)C(N2CCN(C(C3(O)CCSC3)=O)CC2)=O)ccccc1Cl Cc1cc(=O)cc(CNC(c2conc2C(C)NC(c2cnnn2C)=O)=O)[nH]1 C1(CNC(c2c(OC)nsc2)=O)C(C)CCN1C(=O)Cc1csnn1 C1(C(=O)NC(CCCC)(C)C)C2CC3C(C2NC(=O)CCC2CCC(C)O2)C13 N1(C(c2cnccn2)C(=O)NC(C(=O)OC)C)CCN(CC(F)(F)Cl)CC1 c1(C(N(C(CNC(c2ccnc(C)c2O)=O)C)C)=O)cccc2nccnc12 C=CCCCC(C)(C)C(=O)NCC(O)CNC(c1cccc(CN(C)C)c1)=O C1(C(=O)NCC#CCNC(=O)C(F)C(F)(F)F)CC2(CCCC2)CO1 O=C(C1=CCCCCC1)NCC1(C(=O)NC23CC2COC32CCC2)CC1 N1(C(=O)CCC(F)(F)F)CCC2CCCN(C(c3ccnc(CO)c3)=O)C2C1 CC(O)(C(=O)NC1CCCCCN(C(=O)CCn2cnnn2)C1)C(F)(F)F N1(C(c2ccc(COC)o2)=O)CC(C)(C)CC1CC(N1C(C(=O)OC)CC1C)=O Cc1scc(C(=O)NC(C)(C)CN(C(=O)CNC(=O)C(F)(F)F)C)c1C CC(CCN)CC(C)NC(c1c(F)cccc1F)CC(=O)O C=CCC(C)(CC=C)NC(=O)CCC1CCN(C(C2CCC(=O)O2)=O)CC1 c1(C(N2CCC(N(C(CCCOCC=C)=O)CC)C2)=O)cccc2ncoc12 C1(CNC(C(C)C#N)=O)CN(C(=O)C(C)(C)c2ccccc2)CC1N(C)C c1(C(=O)NCC(=O)NCC(=O)NC(C2CCCCC2)CC)ccnc(O)c1F C1(CCCCNC(CCC=C)=O)CCCN(C(c2cc(C(C)=O)cn2C)=O)C1 Cc1nncn1NC(=O)C1CC(CNC(=O)CCOCCOC)C1.C1CC1 c1(SC(C(=O)NC2(CNC(C(CCC)O)=O)CCOC2)C)nc2ccccc2[nH]1 Cc1ccc2oc(C(=O)NCC(C)NC(c3cc4cc(Cl)ccc4o3)=O)cc2n1 C=CCC(C)(C)CC(=O)N(C1CC(NC(c2cnc(O)c(F)c2)=O)C1)C c1(N2CCC(CN(C(=O)CCC3CC(F)(F)C3)C)CC2)ccn2nccc2n1 CC1C(NC(C2C3COCC23)=O)C(C)CCN1c1ncc2ncnc-2[nH]1 c1(OCC(N2CC(N(C(C(C)CC3CCC3)=O)CC)C2)=O)ccccc1[N+](=O)[O-] C1(NC(C(C)(C)F)=O)CC2CC(C1)N(C(c1ccc(CC3CC3)cc1)=O)C2 N1(Cc2c(OC)cc(Cl)cc2)CC2(CCC(C(=O)NCCOC(F)(F)F)O2)C1 c1(C(=O)NC(CC)CN(C(=O)C2=CCCC2C)C)cn2cnnc2cn1 N1(CC#C)CCCC1CNC(=O)NCCOC1(C#N)CC1 C1(NC(c2cc(CC)[nH]n2)=O)CCN(C(=O)C=CC2CCCC2)C(C2CC2)C1 Cc1ccc2nonc2c1S(=O)(=O)N1CCN(C)CC1C(C)C C=Cc1cncc(C(N2CCC(CNC3CC(=O)N(CC)C3C)C(C)C2)=O)c1 N1(C(C(COCC)n2cc(CCCC(C)O)nn2)=O)CCNC(=O)C1CCOC N1(C(C(C)OC)=O)CCCCC12CCCN(C(=O)C(C)OC)C2 c1(C(N2CC(OCCOC)C2)C(=O)NCc2cccs2)nn(CC)nc1Br.C(C)C c1(C(N(CC(C)O)CCNC(CC(C(C)C)O)=O)=O)cc(=O)c2ccncc2o1 c1(C(=O)NCC2(F)CC(CNC(c3cc(CC)no3)=O)C2)ccc(F)cc1C C1(C)(Nc2cc(NCC(c3cccc(Br)c3)(C)C)ncn2)CCS(=O)(=O)C1 CCC(CC(=O)N(CC(N1CCN(C2CC2)C(C)C1)=O)C1CCC1)C(F)F Cc1cc(NC(C2(NC(c3cc4n(n3)CCO4)=O)CCC2)=O)ccc1Br CCCCC(=O)C(=O)N1CCC(C(C)C(=O)NCC2CCCC2)C1 CCCC(C)(C)CC(=O)NC(C)(C)CNC(=O)CN1C(=O)NC(C)(C2CC2)C1=O c1(C(=O)NC(C2CC(NC(C3CCSCC3)=O)C2)C)ccnc(C(C)(F)F)c1 C(=O)(CCCCCCC(C)C)NCC(C(C)C)NC(C(C)OCC=C)=O C12(C(=O)NCC3CN(C(C)C)C3)CC(CN(C(=O)CCC3CC3)C1)C2 C1(c2n(C)ccn2)NC(=O)CCC1NC(C1(C)CCCC1(F)F)c1nnnn1C N1(C(C(CC)N(CC)CC)=O)CCC(C)CC1C(N1CCN(C(=O)CO)CC1)=O c1(CC)c(C)sc(NC(C2(F)CCN(C(C3CCC3)=O)C2)=O)c1C(=O)N(C)C C1(CNC(c2ncn(C(C)C)c2)=O)CN(C(=O)CSC(F)(F)F)CC1O c1(C(=O)NCC2C3N(C(C=CS(C)=O)=O)C(CC3)C2)cc([N+](=O)[O-])cnc1O c1(C(N2CC3(CCN(C(C4(C)CC4(F)Cl)=O)C3)C2)=O)cncc2nc(O)[nH]c12 CCC(CC(C)CO)NC(=O)C(=O)NCC(N1CCC(C)CC1)c1cccs1 c1(C(=O)NC2(C)CC(NC(c3c(C)nco3)=O)C2)ccc(OC(F)(F)Cl)cc1 c1(C(=O)NCCN(C(=O)CC2CC(C)(C)CO2)C(C)C)cc(C2CC2)n(C)n1 C1(NC(CC2ON=C(C)C2)=O)CCCCCN(C(=O)CN2CCCS2(=O)=O)C1 N1(C(CCc2ccn(C)c2)=O)CCN(C(C2CC(S(N)(=O)=O)C2)=O)C(CCO)C1 N(C1CCCc2ccoc21)C(C1OCCN(C(c2c(COC)cco2)=O)CC1)=O CC#CCCCC(=O)N1CCOC(CN(C(=O)C(c2cncn2C)O)C)C1 N12CCC3(CC1)CC3C2=O.c1(C(=O)NC2CONC2=O)noc(CSC)n1.C(C)(=O)O c1(C(N(CCC2CCN(C(C(C)OC)=O)CC2)C)=O)ccc2[nH]c(=N)oc2c1 C1(C(=O)NCC(C)(CO)NC(c2ccsc2C#N)=O)CC(S(C)(=O)=O)C1 N1(C(c2ccc(OC)cn2)=O)CCC2(CC1)OCCC2NC(c1ccccn1)=O c1(C(N2CC3=C(C2)CN(C(C2CCN4CCC2C4)=O)C3)=O)nc2ccccc2[nH]1 c1(OC)ccnc(CCNC(c2cnccc2C)c2nnnn2C2CC2)c1 N1(C(C(C(C)C)SC)=O)CCC2(C1)CN(C(=O)CC1COC(C)(C)CO1)C2 N1(C(Cc2c(C)con2)=O)CCC(NC(c2cnc(Cl)cc2Cl)=O)C(C)C1 CC1CC(NC(c2ccnc(OC3CCC3)c2)=O)CCN1C(c1cscc1F)=O CC1=C(C(=O)NCC2C(C)CCN2C(=O)Cn2ncc(C)cc2=O)CCO1 C1(N)(c2cn(C3CCC(CC(=O)NCc4cnc(CC)s4)C3)nn2)CCOCC1 CN(C)S(=O)(=NS(=O)(=O)NNc1cccc(Oc2ccccn2)c1)C1CC1 c1(CNC2(C(=O)NCCNC(c3n(SCC)ccn3)=O)CC2)ccc(OC)cc1 C1(NC(C(C)OCCC=C)=O)CCC(O)CN(C(c2ccncc2)=O)C1 Cc1ccc(OCCC(=O)NC(C)C(C)(C)NC(C2C=CCC2)=O)cc1 Cc1csc2cc(C(N3CCCC(O)(CNC(C4(O)CC(F)(F)C4)=O)C3)=O)[nH]c12 c1(CC)cc(F)ccc1C(N1CC(NC(C2(O)CCC2)=O)CC(F)C1)=O c1(CN(CCCNC2(C(=O)NCC)CC2)C)ccc(OC)c(C#N)c1 C1(CNC(c2n(C)c(=O)ccc2)=O)CC2CCCCC2N1C(=O)CSC(F)F C1(C(=O)NC2C(CNC(C=C(COC)C)=O)CC2)COC(Cn2cccn2)C1 n1(CC(=O)Nc2c(C(=O)OC)nc[nH]2)ccc2nc(O)nc(O)c12 C1(CNC(CC2C(C)(C)C2)=O)N(C(C2CC3(CCCC3)C2)=O)CCCC1(C)C C1(NC(Cc2c(C)noc2)=O)CC(CO)N(C(c2ncc(Br)cn2)=O)C1 C1(NC(CC(C)C)=O)CC(C)N(C(c2cnc(OC(C)C)cn2)=O)C1 Cc1ccnc(C(=O)NCCC2CCC(NC(=O)Cc3cnns3)C2)n1 Cc1nc2ccc(C(N3CC(NC(=O)CN(C)S(N)(=O)=O)CC(F)C3)=O)cn2n1 Cc1cc([N+](=O)[O-])cc(C(=O)NCC2N(C(c3cnoc3)=O)CCCC2(C)C)n1 Cn1nnc2cc(C(N3CCCOC(CNC(=O)C=C4CCSCC4)C3)=O)sc12 c1(C(=O)NC2C(CNC(c3c(C)cccn3)=O)C2)sccc1S(=O)(=O)C(F)F c1(OC)cc2c(cc1C(=O)NCC1(C)CCCN(C(=O)CCCC#N)C1)CCC2 N1(C(C(CCC)CCC)=O)CCOC2(CCN(C(=O)C(C)(CC)CC)C2)C1 Cc1noc(-c2cn(CC(=O)Nc3cc(C(=O)O)cs3)cn2)n1 C=CC(O)C(=O)N(C)CCOCCCNC(=O)CNC(C1(CC)CCOC1)=O N1(C(CSCCC#N)=O)CC2(CCCC(CNC(=O)CC3CCC3)O2)C1 CC1C(=O)N(C(C2CCCC2)=O)CCN1CSN1CCC2(N)CC2C1 CC1COc2ccccc2CN1C(c1cccc(C(N)=O)c1F)=O c1(N(C)C)c(NC(C2CSCN2C(c2cc(O)ncn2)=O)=O)cccc1Br C1(CN(C)C)COCC1NC(=O)CN(C(=O)CCc1nc(=N)[nH][nH]1)C1CCC1 C1(CCC(=O)NC(C2CCC2)C2CCC2)CCN(C(C2C=CCCC2)=O)C1 C(=O)(C(C)C(C)C1CCCCC1)NC1CC(NC(c2ccc(CCC)s2)=O)C1 C(=O)(C1CCc2nccn21)N1C(CC(=O)N(C)Cc2ccsc2)CC1 N1(C(C(c2ccn(C)c2)C)=O)CC2(CCN(C(c3cnc4c[nH]nc4c3)=O)C2)C1 Cc1cc(F)c(C(=O)NC2CC2CNC(=O)CCCOC(C)C)cc1F N1(CC(=O)Nc2nc(-c3ccccc3F)cs2)CCCCC2CCCCC12 C(CCC(=O)N(C1CC1)CC1CCOC1)(C(C)C)NC(C(CCC)=CCC)=O N1(C(C2(C)CCC2)=O)CC2CC2(CNC(C2C3CCC2(c2ccccn2)C3)=O)C1 c1(C(N2CCC(C(N(CC#C)C)=O)C2CC)=O)cccc2cncn12 c1(CNC(N2CC(Cn3cc(I)cn3)C2)=O)nnc2n1CCS2 CCCC(C(=O)OC)C(=O)N1CCCN(C(=O)Cc2cc(C)on2)CC1 Cc1snnc1C(=O)NCCOCCOCCNC(=O)C(C)CC1CC1 CN1CCC(C(=O)NCCCC2CCCN2C(C2CC(O)C2)=O)c2ccccc21 C(C(O)C(F)(F)F)NC(C1(CCNC(=O)Cn2cncn2)CC1)=O C(C)(CCC(=O)NCCC1CCCOC1)NC(CC1CC(=C)C1)=O N1(C(C(C)(CO)OC)=O)CC2CC(C1)C(CO)C2NC(C1(C(F)F)CCCC1)=O c1(CC(=O)NCC(CNC(CC(C=C)(C)O)=O)O)csc2c(Cl)cccc12 N1(C(c2c(C)occ2)=O)CCOC2(C1)CN(C(=O)C(C)OCCC(C)C)C2 C(=O)(C1Cc2ccccc21)NCC(CNC(c1cc(Cl)cc(C)c1O)=O)OC N1(C(C2C(C=C)OCC2)=O)CCOCCC1C(NCP(C)(C)=O)=O c1(CC(=O)NC(C(C)(C)C)CNC(=O)Cn2cccn2)nc2c([nH]1)CCCC2 C1(C(N2CC(OC(C)=O)C2)=O)(COC)CN(C(=O)C(C)Cc2cnco2)C1 C1(C(=O)NCCCN(C(C)C)C)CC2CC2N1C(C12C=CC(CC1)C2)=O Cc1ccc(C(=O)NCC2CCC2NC(C2CCSCC2)=O)nc1 Cc1c(C(=O)NCC2C(C)CCN2C(=O)CNS(N)(=O)=O)c(C(F)(F)F)nn1C C(=O)(C(F)(F)CCCC)NCc1ccc(C(N2CCOCC(=C)C2)=O)cn1 C1(C)(C(=O)NC(CN(C(c2c(OCC)n[nH]c2)=O)C)C)CCC(=O)N(C)C1 C1(NC(CCCOCCC)=O)CC2(C1)CN(C(=O)CCC(C)c1ccccc1)C2 C1(CNC(C(C)O)=O)(NC(C2CCC(c3cc[nH]n3)O2)=O)CCC(F)(F)CC1 c1(OCC)ccccc1C(=O)O.c12ccc(cc1)-n1cc(nn1)C1(CC1)NC2 c1(CC)ccc(CNCC2(NC(c3cc(F)cc(F)c3)=O)COC2)c(O)c1 C(=O)(C(C(C)O)NC(=O)C(C)O)NC(COC)C1(C)CC1 CCCC(C(C)(C)C)NC(C12C(NC(c3ncccc3C)=O)C3CC1C2C3)=O c1(NC(C2N(C(Cc3ccc(C)nc3)=O)CC(F)(F)C2)=O)ccn2nccc2c1 C(=O)(CCCCC(C)C)N1CC2CC(CNC(c3c(SC)cccc3)=O)C2C1 c1(OC)cccc(C(=O)NCC23COC(CNC(C4(C)CCOC4)=O)(C2)C3)c1 C(CCC(=O)NC1CC(C(F)C(=O)NCCS(C)(=N)=O)C1)OCCOC CCC(c1ccccc1)=CC(=O)NCCC(O)CNC(c1cnns1)=O N#Cc1cccc(C(F)(F)C(=O)OCC2CCC3(COC3)O2)c1 Cc1ccc(Cl)c(C(=O)N(CC(C)CNC(=O)CC2CCN(C)C2=O)C)c1 c1(CNC(C(=O)NC(c2ccccc2)COC)=O)ccc(C2(C(=O)O)CC2)cc1 Cc1ccc(C)c(C(=O)NC(C(=O)NC2(CO)CC3(CCC3)C2)c2cccs2)n1 CC1CN(C(=O)Cc2cccs2)CC(C)N1C(C1(O)CN2CCC1CC2)=O C1(C(=O)NC(C2CCCC2)CNC(=O)CC2CC2(F)F)CC(F)(CO)C1 C(CC(C)(C)CC(=O)NC1COCCN(C(=O)CCc2scnc2C)C1)OC S(=O)(=O)(C1CC1)NCCNC(=O)NC1(NS(=O)(=O)C2CC2)CC1C(=O)O C1(CC(N2C(C(CNC(C(F)=CCC)=O)(C)C)CCC2)=O)CCCC(C)(C)O1 C1(NC(c2cccn(C)c2=O)=O)CCC2(CC1)CN(C(=O)C=Cc1ccsc1)C2 C(N=c1ccn2c(Br)cnc2[nH]1)C12OCC(CNC(CS(N)(=O)=O)=O)(C1)C2 CC1CCN(C(=O)CCCCCN(C)C(C2CCC(C)(C)C2)=O)CCS1 n1(C(C)C)cc(CNC(c2cc(CNC(c3ccco3)=O)no2)=O)cn1 CC1CCCCC1n1nc(-c2cnn(C)c2)nc1-c1ccc(Br)o1 CC(C)C(C(=O)N1CCN(CCF)CC1)C(C)NC(c1c[nH]c(C(N)=O)c1)=O C12(NC(=O)CCCC3CCC3)CC1CN(C(c1sccc1-c1ccccc1)=O)C2 c1(CC)ccc(Cl)c(C(=O)NC2CN(C(C3CCOC3)=O)CC23CC3)c1 c1(C(N2CCC(N(C(C(CCOC)C)=O)CCO)C2)=O)cc(OC)c(O)c(Cl)c1 Cc1cc(-c2noc(C(C)NC(C3ON=C(C(=O)NCC(=O)O)C3)=O)n2)ccc1O c1(OCC)nc(C)ccc1C(=O)NC1CN(C(=O)C=CSC)C1 c1(C(N2C(CNC(Cc3cc(CC)no3)=O)CCC2)=O)nc(Br)cnc1N c1(NC)ccc([N+](=O)[O-])cc1C(N(CCCNC(c1c(OC)cccc1)=O)C)=O c1(C(=O)NC2CCN(Cc3ccc(OC)c(F)c3F)C2)cnc2sc(C)nc2c1 Cc1ccc2sc(C(N3CC(CNC(=O)C(C(C)C)N4CCCC4)C3)=O)cc2c1 c1(N(CC(CCC)O)C)ccc(S(=O)(=O)NC2CCOCC2OC)cn1 C1(C(C)C)CC(CC(=O)NC2(C)CCN(C(=O)C=CC(=O)NC3CC3)C2)CCO1 c1(CN2C(COC(C3CC(C4CC4)=NO3)=O)CC2)cc2c(cc1[N+](=O)[O-])OCO2 N1(C(CN(C)C(N)=O)=O)CCCCC1CNC(=O)Cc1ccnn1C1CCCC1 c1(N2CC(NC(=O)C(C)(C)C3CC3)CC(C)(C)C2)ccc([N+](=O)[O-])c(C#N)c1 c1(C(=O)NC2CC3(CC(CNC(=O)Cc4ccsn4)C3)C2)noc2ccccc12 c1(OC(C2C=CCCC2)=O)ccc(Br)cc1Oc1ccncc1 N1(C(=O)CSC2CCCCO2)CC(NC(C2(CO)CCC2)=O)CC12CCC2 Cc1nn(C)c(F)c1C(=O)NCCC1CN(C(C23CCN(CC2)CC3)=O)C1 c1(C(=O)NC(C)(CNC(c2cc(CO)[nH]n2)=O)CO)[nH]c2ccccc2c1Br N1(C(c2c(CC)c[nH]c2)=O)CCCC1(C)CNC(=O)CC(=O)NC1CC1 N1(C(C(C)C#N)=O)CCN(C(c2cn(C)cc2C(F)(F)F)=O)CC(CO)C1 Cc1c(C(N2CCCCC2CN(C(=O)C(C)n2cccc2)C)=O)ccc(F)c1F C1(C(=O)Nc2ccc(SC)cc2)(OCCNC(=O)CC2CC2)CCC(F)(F)CC1 Cc1nc2nccc(C(N3CC(NC(c4csnc4C)=O)CC3C)=O)n2n1 C(=O)(C(C)(C)CC(=O)NCC1CC(O)CN1C(c1nccc(OC)c1C)=O)OC CCC(C)(C(=O)NCC1CCC(NC(=O)C(C)O)C1)OC c1(C(N2CCC(O)(C(=O)Nc3c(C#N)n[nH]c3)C2)=O)cc([N+](=O)[O-])c(O)cc1O Cc1cc(C(N2CCC3(CCC3)C2)=O)ncc1-c1cnc(C(=O)O)cc1C C12(CNC(C3(C)CC4CC4C3)=O)CCC(CC1)N2C(=O)COCC1CCCO1 C1(N(C(=O)CCc2cccs2)C)CCCN(C(C2(CCO)CC2)=O)CC1 C1(NC(C(CC)(C)C)=O)COC2(CCN(C(=O)C(F)(F)c3csc(C)c3)C2)C1 c1(C(N(CC(C)NC(CC2N(CC)CCC2)=O)C)=O)c(Br)ncn1C C#CC1CC2(CC(C(N3CCOCC3CNC(=O)CN(C3CCSC3)C)=O)C2)C1 c1(OCC)ccc(C(N2CC(CO)(NC(=O)CC3CCCC3(F)F)C2)=O)cc1C c1(C(C)=O)ccc(C(=O)NC2CCC(CNC(C3NC(=O)CC3C)=O)CC2)cn1 CCC(C)(C(=O)NCC1(F)CC(CNC(C2(C)CCCS2)=O)C1)C(N)=O C1(NC(Cc2cc(CC)no2)=O)CCN(C(=O)C=Cc2ccccc2Cl)C1(C)C C12(OC)CC(C1)N(C(=O)C(=O)NCC1CCC(C(F)F)CC1)C2 c1(NC(CNC(CN2CCN(S(C)(=O)=O)CC2)=O)=O)nccc(Cl)c1Cl Cn1ccc2ccc(C(N3CCC(NC(=O)Cc4nc(=N)[nH][nH]4)C3)=O)cc12 C1(C(=O)NOCCOCCO)CCN(C(=O)c2n[nH]c3c2COC3)O1 c1(NC(C(C2CN(C(C3CCC(CC)O3)=O)C2)O)=O)cnc2ncnn2c1 C1(CNC(CC2(CSC)CC2)=O)CCCC2(CN(C(=O)CC(C)CF)C2)O1 N1(Cc2ccc(C#C)s2)CCC(O)(C(=O)NC2CCC(C)CC2)CC1 c1(C(=O)NC(C)CNC(=O)CSCc2ccncc2)ccc2nc[nH]c2c1 C(C(=O)NCCN(C(c1cnc(C)nc1C)=O)C(C)C)(C(C)(C)C)NC(C)=O N1(C(C2C(C)C2)=O)Cc2ccnn2CC(NC(c2ccn(C3CC3(F)F)n2)=O)C1 c1(C(=O)NCC2(O)CCCN(C(CCSCC(C)C)=O)C2)cc2cnn(C)c2s1 c1(OC)ccc(C2CN(C(C3(S(C)(=O)=O)CCC3)=O)C2)c(Cl)n1 CC(CC(=O)c1cccc([N+](=O)[O-])c1)C(=O)N1CC2(C(=O)O)COCCC12 CS(=O)(=O)c1ccc(CCN=C(NCCF)NCCC(O)C(F)(F)F)cc1 C1(NC(c2nc(C(C)C)sc2)=O)CCCN(C(C23CC(CC(F)F)(C2)C3)=O)CC1 c1(C(N2CC(NC(C(CC)n3ccnc3)=O)C(C)C2)=O)ccc(C(C)C)nc1C c1(C(N(CCCNC(C2(C#N)CCSCC2)=O)C)=O)cc2ccncc2[nH]1 N1(C(C(C)SC(C)C)=O)CCC2(NC(=O)CCS(N)(=O)=O)CCCC12 c1cc(-c2ncccc2N=[N+]=[N-])c2c(c1)NCCO2 n1(CC=C)cc(C(N2CC(NC(C3CC3c3ccsc3Br)=O)C2)=O)nn1 Cc1cc(C(N2CCC23CN(C(c2cc(Cl)cnc2Br)=O)C3)=O)nc(Cl)c1 c1(NCC(C)CNC(c2cccnc2-n2cccn2)=O)nc(Cl)[nH]c2ncnc1-2 C1(C(=O)NCC2CC(NC(CCSCC)=O)C2)COc2ccc(Cl)cc2O1 c1(OC(C)C(=O)NCCCNC(=O)CN2CCCNS2(=O)=O)ccc(F)c(F)c1 C12(CC(=O)NC3CCCC(NC(C(CSC)O)=O)C3)CCC(CC1)OC2 C12(CNS(C(CCC)C)(=O)=O)CCC(C#N)(CO1)C2 c1(C(=O)NCc2cn(-c3ccc(C)nc3)nn2)cc(C)cc2ccoc12 C1(NC(CSCC(=O)OC)=O)CC(NC(=O)C(C)OC)C1 c1(SC)cc(N2C(C(=O)NC(c3ccccc3Cl)C)CC3CC23)ncn1 CCC(CC)C(C(=O)Nc1ccccc1)N1CCC(C)(Cc2ccccc2)CC1 C(=O)(CCCS(C)(=O)=O)NC1C2N(C(C(NCP(=O)(O)O)C3(C)CC3)=O)C(CC2)C1 C1(NC(c2c(C)nn[nH]2)=O)CCN(C(C2(F)CC3(CCC3)C2)=O)CC1CO N1(C(C2(C)C=CCCC2)=O)Cc2ccccc2C(NC(C2CCCCCC2)=O)C1 C1(O)(CNC(CCC(=C)C)=O)COC2CC1C2 c1(C(N2CCC(C(C)NC(C3CCC34CCC4)=O)CC2)=O)ccc(S(C)(=O)=O)[nH]1 c1(N2CC(NC(c3cc(SC)oc3)=O)CC3(C2)CC3)ccc([N+](=O)[O-])c(O)n1 c1(NC2CC(NC(c3cc(CO)ccn3)=O)C2)c(O)cc(C(=O)OC)cc1O Cc1cc(O)cc(C)c1CC(=O)NC1CC(NC(C2CN(CC(F)(F)F)C2)=O)C1 CN1C(=O)c2ccccc2C1C(=O)NCC1CC2(CO1)CN(C(=O)C=C(Cl)Cl)C2 c1(CNC(C(=O)N(C(C)C)C)C)c[nH]nc1Br c1(NC(C2CCCN2C(=O)C(c2ccccc2)O)=O)nc(Cl)ccc1O N1(C(CC(C)NC(CC(=O)NC(C)CC2(O)CCOC2)=O)=O)CCN(C)CC1 c1(N(CC(C)N(C(C)=O)C)C)nc(=NC(C)c2ccc(C)o2)[nH]c2c1COCC2 C1(OC)CC(F)CN(C(C2COC(CNC(=O)CC3CCC3)C2)=O)C1 c1(C(N2CC(NC(c3c(SC)cccn3)=O)C2)=O)c(N)c(C(F)(F)F)nn1C C1(CC(=O)NCCOCCC(C)C)CN(C(C2NC(=O)OC2C)=O)CCC1C c1(N2CCC(CN(C(Cn3cc(CC(C)(C)O)nn3)=O)CC)C2)ccc(F)cc1F CC(C)C(F)C(=O)N1CCN(C2CCN(c3cc(C(C)(C)C)ncn3)CC2)CC1 Cc1ccc(-c2cccc(C3CC3C(N3CCC4(CCOC4)C3)=O)c2)c(F)c1F C(=O)(CC(CN(C)C)C(F)F)OCc1cc(C)ncn1 N1(C(c2n(CC)ccc2)=O)CC(CNC(C2CCCC2F)=O)CCC1C CC(C)C(O)C(=O)N(CCNC(=O)CCc1ncc[nH]1)CCOCCO Cc1nc(=NC(=O)CC2CCCN2Cc2cccc(C#N)c2Cl)s[nH]1 N1(C=O)CCC2C(CCCN2c2c(CC)nc3sc(C)cn32)C1 N1(C(C)=O)CCN(C(C2CCCN2N=O)=O)C(c2cccc(Br)c2)C1 c1(NC(C2CCN(Cc3c(C)nc(F)cc3)C2)=O)cccc2nc(O)[nH]c12 Cc1c(C(=O)NC2CCCCC2N(C(=O)C(C)c2ccco2)C)sc2ccsc12 C1(C(C)C)CN(C(=O)CC(C)NC(=O)C2CC2)CCN1C(c1occc1F)=O C1(CC=C)(C(N2CCC(n3ccnc3)C2)=O)CCN(C(=O)CC(C)(F)F)C1 N1(C(c2nc(C(C)C)sc2)C(=O)NC2(C)CC2)CCC2CC2C1 c1(C(=O)NCC2C(NC(C3(COC)CC3)=O)CCCC2)c(C)nc(=N)[nH]c1C c1(SCC(C)C(=O)N2CC(N(C(=O)CCN3CCOCC3)C)C2)ccc(F)cc1 c1(C(N2CC(OCC(=O)N(CCCC)C(C)CC)C2)=O)ncccn1 N1(C(CC(C)O)=O)CC2CCC1C1CN(C(c3cccnc3C(N)=O)=O)CC21 c1(C(=O)NC(C(C)NC(=O)CN(C)C(N)=O)C)c(Cl)cncc1Br C1(CCO)(OC)CN(C(=O)COCCOC(C(=O)NCC(C)(C)O)C)C1 CCC(C)C(C(=O)NCCn1ccnc1C(=O)O)c1ccccc1 c1(C(=O)NC2CCC(NC(C(C)(C)F)=O)C2)cc([N+](=O)[O-])ccc1SCCO c1(OC)ncc(C(N2CC(NC(c3cnc[nH]3)=O)CC2(C)C)=O)cc1C(F)(F)F CCCC(C)(CO)NC(=O)NCc1ccc(COC)cc1 C(=O)(CC(CC)C(F)F)N1CCN(C(c2cnc(CCC)s2)=O)C(CCC)C1 c1(C(N2CC(NC(C=CC(CC)=CC)=O)C2)=O)ccnn1-c1ccncc1 C1(CNC(CCC)=O)CN(C(=O)C(C(C)C)OCC(C)C)CC12CCC2 C(=O)(CC(C)P(C)(C)=O)N1CC(CCNC(C(CC=C)(F)F)=O)C(C)C1 c1(C(=O)NCC2C(NC(CSCC#C)=O)CCCC2)ccc2c(c1)NC(=O)CC2 C(N=c1cc(C)c(C#N)c(C)[nH]1)C1N(C(c2cnc(OC)c(C)c2)=O)CCCC1 C(=O)(C1=CCC2(COC2)OC1)N1CC(CNC(CNC(CCC)=O)=O)C(O)C1 C(=O)(C1=CCN(C(C2(NC(C)=O)CCC2)=O)C1)NCc1c(CC)noc1 C1(NC(CCN(CC)CC)=O)C2CC(NC(C3CCOC3(C)C)=O)CC12 N1(C(=O)NC2C(C(C)C)C3CCC2C3)CC2CC1C1OCCOC21 C=C=CC(C)C(=O)N1CC(COC)(NC(c2cc(C)n(C(C)CC)n2)=O)C1 c1(C(C)F)ccc(C(=O)NCC2(F)CCN(C(=O)C#CC(=O)N(C)C)C2)cc1 C1(NC(c2c(C)n[nH]c2)=O)CC(NC(C2CC23CCCC3)=O)C(O)C1 c1(C2(OC(C3(C(N(C(=O)CC4CC4C(F)(F)F)C)=O)CC3)=O)CC2)ccccc1 C12(NC(=O)Cc3ccon3)CCCC1N(C(c1cc(C(F)(F)F)ncn1)=O)CC2 N1(C(C2=C(C)OCC2)=O)CCC(C(=O)Nc2cnn(C)c2C)CC1(C)C c1(CC#N)cc(Br)ccc1NC(C1CC(F)CN(C(=O)C2=CCCC2)C1)=O C1(C)(CCNC(C)=O)CCN(C(=O)CNC(CC(CC)SC)=O)CC1 n1(C(C(=O)N(CC(C)(C)OC)C)C)cc(-c2ccc(Cl)s2)nn1 c1(OC)cc(C(=O)NC(C)(C)CNC(C2CC3CC2C3)=O)ccc1OC(F)F c1(C(=O)NCC#CCNC(C2(C#N)CC3(CC3)C2)=O)cnc2c(c1)COCC2 N1(C(c2cc(C)n(C)n2)=O)CCCC(NC(=O)CCC2CCC(=O)N2)CC1 Cc1ccc2[nH]c(C(=O)NCC(CNC(=O)C=CC(C)(C)C)CO)cc2c1C C1(NC(C(CCC=C)(F)F)=O)CC2CN(C(=O)CCC(N)=O)CCN2C1=O C1(NC(C(N2CCOC2=O)C)=O)CCCN(C(C2CC=CCC2)=O)C1 C1(NC(c2c(N)nccn2)=O)CN(C(=O)CC2=CCCC2)CC12CCCC2 Cc1nc(CNC(c2cc(CO)n(C)n2)=O)oc1C(=O)NCC1CC1C Cc1ccc(OCCC(=O)NCC(CNC(=O)C2=CCOC2)CCSC)cc1 c1(C(=O)NCC2(CN(C(c3nc(C#C)sc3)=O)C)CC2)cc(C)c(Cl)cc1OC c1(C(N2CCC(C(=O)NC3CC4CCC(C3)N4)C2)=O)cccc(Cl)c1F c1(C(N2CC3C(C(=O)Nc4ncc(C)s4)(C3)C2)=O)cc2ccc(Cl)cc2nn1 C(=O)(C1=NOC(C)(C)C1)NCCCOCCC(=O)NC1(CC=C)CCCC1 O=C1CCC(S(=O)(=O)N2C3CCC2CC(NC(c2cc(I)ccc2O)=O)C3)CC1 c1(C(=O)OCC(=O)N(c2ccc(OC)cc2)C(C)C)cc(F)c(C=O)cc1F C1(C(N2CCC(N(CCCC)C(C3CC=CCC3)=O)CC2)=O)COCCC1(F)F CC1CCCC(C(N2CCN(CC3CN(C(c4ccnnc4O)=O)C3)CC2)=O)C1 N1(C(c2cnc(SC)s2)=O)CC(C)(CNC(C2CC3(CC3)CO2)=O)CC1(C)C Nc1cc2[nH]c(O)nc2cc1C(=O)NCC1CN(C(C2CC2(Cl)Cl)=O)CCO1 C=C=Cn1ccc2c(N3CCC(C)C(C)C3)ncnc12 c1(OC(C)C)ccc(F)c(NC(c2ncoc2-c2ccccc2)=O)c1 Cn1cc(CC(=O)NC2CC2CNC(c2ccc(C(C)(C)C)s2)=O)cn1 c1(CC(N2CCCC(C3N(C(COC)=O)CCC3)C2)=O)c[nH]c2c(F)cccc12 c1(C(=O)NC(C)C(c2ccccc2)NC(=O)CC2CCC2)ccnn1C(F)F N1(CCNC(C2(n3ccnn3)CC2)=O)CCc2cc(F)c(F)cc21 CC(CC(=O)NC1CC(CC(=O)NC2CCC(N=[N+]=[N-])CC2)C1)C(F)(F)F c1(C(=O)NCCN(C(CCC#C)=O)C2CC2)cc2ccccn2c1 C1(NC(c2c(C(F)F)cccc2F)=O)CC2CCC1N2C(C1(O)CC1)=O O=C(CCCCC(F)(F)F)NCC1CCCCC1NC(C1CCC2(CCC2)C1)=O N1(C(CC(COC)(C)C)=O)CC2(CCN(C(c3nc(C(C)C)no3)C)CC2)C1 N1(C(c2cnc(C(F)F)s2)=O)CCCC(CNC(=O)C(F)(F)c2nccs2)CC1 CC(N=c1[nH]c(=NC(C)C(F)F)c2sccc2[nH]1)c1cncs1 N1(C(c2scnc2C(F)(F)F)=O)CCC2CCN(C(C3CCSC3)=O)C2C1 C1(NC(c2c(C)n(C3CC3)nc2)=O)CCN(C(C2(C)CCCS2(=O)=O)=O)CC1O N1(C(c2cc(C)sc2N)=O)CCC(NC(=O)CCc2ncc[nH]2)C(F)C1 C(C(C(=O)NCCN1CCC(O)C1)NC(=O)C=NOC)OCC c1(OC)cc(N2CCCC(C)C2CNC(c2ccc(Cl)o2)=O)ccc1[N+](=O)[O-] c1(C(=O)NC(C(C)C)CNC(=O)C2=NOC(C(C)(C)C)C2)nn(C)c2c1CCC2 C1(CNC(c2ccc(C(C)C)o2)=O)CN(C(C2C=CCS2)=O)CC1(F)CO CS(=O)(=O)c1ccc(C(=O)NC2CCSC23CN(C(c2ccc[nH]2)=O)C3)c(Cl)c1 CCC(C)C(O)C(=O)NC1(C(N2CCN(C(C)C)C(=O)C2)=O)CCSC1 N1(C(c2ccc(CC(N)=O)cc2)=O)CC(CNC(CC(C)C)=O)CC1C c1(-c2cn(CC3N(C(CC(C)C)=O)CC3)nn2)ccc(Cl)c(N)c1 c1(CN(C)C(C2CCC(C(N3CCNCC3)=O)O2)=O)c(S(N)(=O)=O)cnn1C c1(C(N2CC(C)(NC(=O)CNC(=O)C=Cc3ccco3)C2)=O)nccc2ccsc12 c1(C(C)(C)NC(=O)CCOC2COC2)nc(=O)o[nH]1.C12CC(C1)C(=O)N2 c1(C(=O)NCC2CC3CC(C2)N(C(=O)CC2CCOC2)C3)n[nH]c2c1CCCC2 C(=O)(C(CNC(=O)CN(C1CCC1)C)OC)N1C(C(=O)OC)CC1 C1(CCOC)CN(C(=O)CC2CCCC2C(=O)O)CCN1C(c1ccccc1)=O c1(CNC(C=CC)=O)cccc2c1CCN(C(C1CCOC1(C)C)=O)C2 C1(CC(=O)N(C(C)C(=O)NCC(C)CO)C2CC2)CCCC2CC12 C(C(=O)NC(C)CNC(c1cc(CN(C)C)on1)=O)(C(C)(C)C)OCC n1(C(C)C)ncc(Cl)c1C(=O)N(C1CCN(C(c2ccoc2Cl)=O)C1)C c1(C(=O)NC2CCC(CNC(c3c(C(C)C)nns3)=O)C2)c(F)ccnc1F C1(C(=O)OCC)CCN(C(C2(NC(C3CC3c3nc[nH]n3)=O)CCCC2)=O)C1 N1(c2nnc(C)o2)CCCC(C)(C(=O)NCCOc2ccccc2C)C1 CC(C)C(C)(CNC(=O)Cn1ncnn1)NC(C1CS(=O)C1)=O Cc1nn(C)cc1C(=O)NC1CN(C(C2CCCCO2)=O)CC1C N=c1nc(Cl)cc(C(=O)NCC2CCCCC2NC(C2CC(=O)N2)=O)[nH]1 c1(CC(=O)NC(C)CC2CN(C(c3cncn3C)=O)C2)ccc(Br)c(Cl)c1 c1(OCCC)ccc(Br)cc1CN(C)CC1CCCCN1C(=O)CC1CC12CC2 N1(C(C2(CSC)CC2)=O)CCC(NC(=O)Cn2nc(C)c(C)c2C)C(O)C1 C1(C(=O)NCCc2c(C)noc2C)C(C2CC2)CCN1C(c1sccc1F)=O C#CC1(C(N2CCC(C(C)C)CC2)=O)CCN(C(c2ccn(C(F)F)n2)=O)C1 N1(C(Cn2ncc(C(=O)OC)c2)=O)CCC(NC(c2cc(C)no2)=O)C1C C1(c2n(C(C)(C)C)nnn2)(NCC2(CO)CC3CC3C2)CC2C=CCC12 C12(CC(=O)NCC(CN(C(C(c3cncnc3)C)=O)C)C)CCC(CC1)C2 C1(C(C#C)C)CCN(C(C2CCOCC2NC(c2ocnc2C2CC2)=O)=O)CC1 C(CCCCCNC(=O)Cc1ccnn1C1CCC1)NC(C(=O)NCC)=O C=CC(C)(CC)C(=O)NCCCN(CCCNC(=O)CSCCCNC(C)C)C C1(C(=O)NC(C#C)(C)C2CCOC2)CCCN(C(C2CC=C(C)CC2)=O)C1 C(C1=NOC2CCCCC12)NC(N1CC(CC)OCC1)=O C1(CC(=O)NCCC(C)NC(C2CCCOC2C2CC2)=O)CCN(CCF)CC1 C1(NC(C(C2CC2)OC)=O)CC2CC1N(C(=O)CCC(=O)c1cccc(N)c1)C2 C(=O)(C1=CCCCO1)NC(CCN(C(Cc1cccc(COC)c1)=O)C)C(C)C C12(NC(Cc3c(C)cco3)=O)CCCC1CN(C(=O)CC1(O)CCOCC1)C2 C1(C(N2CC(CC(=O)NCCN(C)C)OCC2)=O)CCC2(CCC2)C1 c1(CNCC2N(C(C3CC(C)OC3)=O)CCC2)cc(O)ccc1N N1(C(C(N2CCC(O)CC2)C)=O)CCOC(C)(CNC(=O)CN(C)C)C1 N1(C(c2cccc(NC)n2)=O)CC2CCC1C(NC(C1CN(C)CC(C)O1)=O)C2 C(=O)(C(C)C(F)(F)F)NC(C)Cn1cc(CNC(C2CCCOCC2)=O)nn1 c1(C(N(CCCC(=O)O)CC)=O)ccc(C2CCC2)cc1 CCCCC(F)C(=O)NC(C1CCCC1)CNC(=O)Cn1nc(C)oc1=O CC1(CNC(C2COCCO2)=O)CCN(C(=O)CNC(=O)CCCCO)CC1 C=CCC(CC)C(=O)NCC1CC(NC(c2cnn(CC)c2C2CC2)=O)C1 N1(c2nnc(-c3n(C)ncc3I)n2CC)CC2(CC(C(=O)NCC3CC3)C2)C1 c1(C(=O)NC2C(C)N(C(C3(C)CCC(=O)N3)=O)CC2)ccc2cc(Cl)ccc2c1 c1(C(=O)Nc2cccc(NC(=O)NCCF)c2)ncc([N+](=O)[O-])cc1Br c1(OC)cc(N2CCC(NC(c3cnn(C)c3)=O)CC(C)(C)C2)ccc1[N+](=O)[O-] c1(N(CC(CN(C(C2(C(=O)NC)CC2)=O)C)O)C)cnc(F)cn1 N1(C(CCOC)=O)CCC2CCCN(C(c3coc4c(C)cccc34)=O)C2C1 c1(CC(=O)N(CCN(C(=O)C(O)C(C)OC)CC)CC)cncc(F)c1 C1(CC(=O)N(C2CN(C3CC3)C2)C)CCCN(C(=O)Cn2cccnc2=O)C1 C(CNC(C1C=CCS1)=O)(CC(F)(F)F)NC(c1cn(C)nc1C(C)(C)C)=O c1(OC)cc(C(N2CC(NC(C3C=C3C)=O)C(C)C2)=O)ccn1 C1(C(=O)OC)CCN(CC2(CO)CCNCC2)CC1.c1(CN)nc(C)no1 C(C)(C(CC(=O)NCC1CC(C(F)(F)F)C1)NC(=O)CC1C=CCC1)OC c1(C(N(C)CC2N(C(c3cc(C)ns3)=O)CCCC2)=O)csc2cncn12 C(c1ccc(C)cc1C)=CC(=O)NCC(CNC(c1scc(C(C)=O)c1)=O)O c1(C(N2CCCC(N(C(c3nnn(CC)c3C)=O)CC)C2)=O)c(F)ccc(F)c1O C1(CC#C)CCN(C(C2(CNC(C3CCC(=O)O3)=O)CCCO2)=O)C1 c1(OC)cc(CC(=O)NCC(CCNC(c2csc(C)c2)=O)OC)ccc1F CC(Cc1ccncc1)(C(=O)O)NCC(CNc1ccccc1)CO N1(C(c2c(CC(C)C)onc2)=O)CCC(NC(=O)C(O)C(F)F)C2(CCC2)C1 C(=O)(C1=CCN(C(c2cnn(C)c2OC)=O)C1)N(C(C(=O)OC)C)C c1(N2CC3(C(C(N4CCC(Br)CC4)=O)C3)C2)ncc2cn[nH]c2n1 CC1CC(C(=O)NC2(CCCCNC(=O)CCN3CCC3)CC2)=NO1 c1(C(C)NCCC#CC)cnc(N2CCOCC2)nc1 c1(C(N2CC(F)CC(C(N(C3CC3)CC)=O)C2)=O)c(Br)ccc(OCC)c1F CCCC(C(=O)N1CCC(C2CCCN2C(=O)C(CC)OCC)C1)S(N)(=O)=O N1(C(C2C(CCC)C2)=O)CC2(CCN(C(=O)C(C)(C)COCC)CC2)C1 c1(C2(C(N3CCC3COCC3CCC3)=O)CC2)cc(F)ccc1F C1(CNC(CC(CC)O)=O)CC2(CC2)CN1C(=O)CN1CC(=O)N(C)C1=O C(C)(CCCCNC(C1(C)CCSCC1)=O)NC(C1(COC)C=CCC1)=O C(=O)(C(C)(CC)CC)NC(CCC)CNC(=O)Cc1cccnc1 C(=O)(C1CCCc2cccnc21)N(CCC(C(C)C)NC(CCOCCC)=O)C C1(C(=O)NCC=C2CCN(C(C3(COC)CC=CCC3)=O)CC2)CCOC(C)(C)C1 c1(C(=O)NCCCN(C(CC=CC)=O)C2CC2)nn(C)c(C2CC2)c1C N1(C(CCc2c(C)noc2C)=O)CCC2(CCC2NC(=O)CC#N)CC1 C1(NC(COC(C)C)=O)(CO)CCCN(C(=O)C(C)CN2CCOCC2)C1 C1(CNC(C(C(C)(C)C)SC)=O)CC2CCC(C1)N2C(=O)CSCC(F)(F)F Cc1ccc2c(=NC3CC(CC4CC4)C3)[nH]c(=NCC3CCCCO3)[nH]c2c1 c1(OC)cccc(-c2cncc(CN3CCCC3C(F)(F)F)c2)c1 c1(C(=O)NC(CN(C(c2cnc(CC)s2)=O)C)(C)C)cc2cncn2c(O)n1 N1(C(c2c(C)n(C)cc2)=O)CCC2(CO)CN(C(C3(S(C)(=O)=O)CC3)=O)CC2C1 c1(CNC(C2CCCN(C(C3(Cl)CCCCC3)=O)C2)=O)cccc(CO)c1 CCC(O)C(F)(F)C(=O)NCC1CC2CCC(C1)N2C(=O)CC1CCS(=O)(=O)C1 N1(CCC(=O)NC2CN(C(=O)CNc3nccs3)CC2O)CCCCC1=O CCS(=O)CC(=O)NCC(C(F)(F)F)N1CCN(C(C2CCCSC2)=O)CC1 C1(NC(=O)C2=CCOCC2)CC2CC1CN(C(c1cnoc1-c1cccs1)=O)C2 N1(C(COCc2cc(C)on2)=O)CCOCC1CCNC(C1CNC(=O)N1)=O C1(C)(C(c2n(C(C)C)nnn2)NCc2ccnc(Br)c2)CCCC(F)(F)C1 c1(OC)cc(CN(C)C(c2ncoc2C2CC2)=O)sn1 CCCC(C)(C)C(=O)NC(CNC(=O)C(O)CCSC)CC Cc1cc(O)cc(=O)n1CC(=O)NC1CN(C(C2(CC(C)C)COC2)=O)CC1O N1(CC(=O)NCC(C#C)CC2CC2)CCN(C(C2(Cl)CC2C(C)=O)=O)CC1 C1(C(N2CCC(CCC(=O)O)CC2)=O)CC2CNCC1C2 N1(C(C(C)(O)C2CC2)=O)CC2CCN(C(=O)C3=NN(C4CC4)C(=O)CC3)CC2C1 C1(C(=O)NCCCC(C)(C)F)CC2(CC(NC(C3CCCO3)=O)C2)C1 CCCC(C(=O)OCC(c1ncc(C)s1)=O)NC(=O)OC(C)(C)C c1(C(N(C)CC2N(C(CN3C(C)CC3)=O)CCC2)=O)ccc(Br)cc1F C#CC(C)(C)C(=O)NC(CNC(c1cccc(C2(C#N)CC2)c1)=O)C(C)(C)C CC1CC(NC(C2CCN(CCF)CC2)=O)CCN1C(C1CCSC1)=O C1(c2nnc(CC)o2)CC(O)CN1C(c1cccc(=O)o1)=O C(=O)(CC(O)CCSc1ccccc1)NCC=CCNC(C1(COC)CCC1)=O CC(C)C(C(=O)N1CC(F)C(F)C1)C(C)NC(=O)COC1CCC1 C1(C(=O)NCC(=C)CCNC(=O)CNS(=O)(=O)CCC)CCC(C)NC1=O C1(NC(c2c(C(=O)OC)cccc2)=O)CC2(CCN(Cc3ncco3)CC2)C1 C(CC(=O)NS(=O)(=O)CC1CCSC1)SC c1(C(=O)NC(COC)CNC(c2cncn2C)=O)cccc(F)c1O C1(C(N2CCN(C(CC)=O)CC2)=O)CC(N=[N+]=[N-])CN1C(=O)CN1CCOC1=O c1(CC)c(C(=O)NC(C)CNC(c2ccc(N)cc2C)=O)cccc1F C=C(C)CC(C)C(=O)NCC1CN(C(=O)Cc2cc(F)ccc2Cl)C(C)(C)C1 c1(C(CNC(C2(C(F)F)CC2)=O)NC(CCC=C)=O)cc(F)cc(Br)c1 N1(C(=O)C(=C2CCCCC2)F)CC(NC(C2(CO)CCCCC2)=O)CCC(O)C1 c1(C(=O)NCC(CNC(c2c(CC)nn(C)c2)=O)O)cnc2cnn(C)c2c1 N1(CCCNC(C2CC(NCc3ccc(C)nc3)C2)=O)CCS(=O)(=O)CC1 C1(C(=O)NCc2cc(C(=O)NC(C3CCCCC3)CC)n[nH]2)CCCCC(=O)N1 c1(C(N2CCC(CC=C)(NC(c3cc(O)no3)=O)C2)=O)cc2c(s1)CN(C)CC2 C(=O)(CCCC(F)(F)F)NC(CNC(=O)CCCN1CCCC1)C1CCC1 c1(-c2cn(C(C(C)O)C)nn2)cnn2c1CN(C(c1cc(C(F)F)no1)=O)CC2 c1(C(N2CC3C(CNC(C4(SC)CCC4)=O)C3C2)=O)cnc2ccoc2c1 N1(C(C(C)N(C(C2(Cl)C(C(C)=O)C2)=O)C2CC2)=O)CCN(C)C(CO)C1 N1(C(=O)Nc2cc(CC)ncn2)CCC2(CCC(OC)C2)C1 C1(NC(C(CSC)OC)=O)CCOCC1C(=O)NCc1nn[nH]n1 N1(C(c2c(NCC)scn2)=O)CCC2(C1)CN(C(=O)C(CC)OC)CCO2 c1(OCC#C)c(OC)ccc(CNCc2ccc(-c3csc(C)n3)s2)c1Cl CC1(C)CCCC1C1CCN(CC2CC3CCC2C3)C1 C(CCC(=O)NC(COC(C)C)CNC(=O)Cc1nc(C)no1)OCCOC c1(N2CCC(SC)CC2)ncccc1S(=O)(=O)N1CCOC(N2CCCC2)C1 C(=O)(C#CC1CCCOC1)NCCCC(C)NC(C1Cc2ccccc2N1)=O c1(C2(NC(c3ccc(C4CCCCO4)cc3)=O)CC2)ccccc1Br CC(C)(C#N)CCC(=O)N1CCN(C(=O)C=Cc2ccco2)C(CCO)C1 CN1CC2(CC2)CC1C(=O)NCC1(NC(c2cccc(F)c2N)=O)CCCCC1 S(=O)(=O)(c1cccnc1NCCOCCO)NC1C(C)N(C)CC1 c1(Nc2nnc(CSc3cccc(OC)c3)o2)ccc(S(=O)(=O)C2CC2)cc1 c1(C(=O)NCCCC(C)NC(c2cccc(C#N)c2)=O)c2c(nn1C)CCOC2 Cc1nc(S(=O)(=O)NCCC(=O)Nc2ccc(F)cc2F)cn1C C(=O)(CC(C)(C)C)N(CC(=O)NCC(=O)NC(C(C)(C)O)C1CC1)C c1(C(N(C2CCN(C(c3cnnc(Cl)c3)=O)C2)CC)=O)ccccc1OC c1(CC)ccc(C(=O)NC(C)(CNC(=O)C(C)(C)COC)C(C)C)nc1 c12nc(C)ccc1C(=O)N1CC=CCC1C(=O)N2.n1(CC)cc(CO)nn1 C(CCCC(=O)NCCC1CSCCN1C(=O)CCc1cnc(O)nc1)OCC C1(NC(c2c(C(C)C)cccc2)=O)CC2CCC(C1)N2c1nc(Cl)ncc1Br Cc1cc(Nc2n[nH]c(C(F)(F)F)n2)nc(C)c1.C1(S)CCC(N(C)C)CN1 N1(C(=O)OC(C)(C)C)CCC(C2(NC(=O)NC3CCC4(CCC4)C3)CC2)C1 c1(NC(C(N)c2cccs2)=O)cccc2c1C(=O)NC2=O CC(c1cccs1)=CC(N1CCN(C(=O)CCC(=O)c2cccnc2)CC1)=O CCC(CC(=O)NC1CCC(CC(=O)N(C2CCSC2)C)CC1)C1CC1 N1(C(CC2N(CC)C(=O)CC2)=O)CCN(C(c2cccc[n+]2[O-])=O)C(CF)C1 N1(C(c2c(C)nc(O)[nH]2)=O)CCC(NC(c2c[nH]c(=O)cn2)=O)CC1C C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NC1CCN(c2ccnc(C)n2)CC1F C1(C(C)NC(C(C2CCCCC2)OC)=O)CCN(C(=O)CC(C)O)CC1 N1(C(N2C(C)CC(CC(=O)OC(C)(C)C)C2)=O)CCOc2ccccc2C1 N1(C(=O)CC2CCN(CC3CC3)C2)CC2CC1CC21OCCO1 C1(C(N2C(CNC(CCC(=C)C)=O)CC3CC32)=O)CCc2ccccc2CC1 CC1(C)C2CCC(C2)C1NC(=O)CCCCNC(C1(CO)CCC1)=O C1(CCC(=O)N(CCN=[N+]=[N-])CC)CCN(C(=O)CCN2CCCC2=O)C1 C#CCC(C)(C(=O)NCCN1CCC(CO)C1)NC(=O)C(F)n1ccnc1 C1(C(=O)NCC2(O)CC(NC(c3cnsc3)=O)C2)CCC2CC2CC1 C1(C(=O)NCCCC(C)(C)C)N(C(c2cccnc2O)=O)CCCC1(C)C N1(C(C2(C)C(C)OCC2)=O)CCC=C(CNC(=O)CCC2(C)CC2(F)F)C1 c1(NCC2(CC)CCOC2)cc(NC(=O)NC)ccc1C N1(C(=O)NCC)CCCc2cc(OCC#N)ccc21.c12ccc(cc1)o2 Cc1ccc(C(N2CCN(C3CCCN(C(C4(F)CC=CC4)=O)C3)CC2)=O)n1C CN1CCN(C(C2(NC(c3cc(F)c[nH]3)=O)CCN(C)C2)=O)CC1C1CC1 C1(COC)CN(C(=O)CN(C)C(N)=O)CCN1C(=O)CN1CC2CC2C1 N1(C(CNC(CCCOCC)=O)=O)CCOC(C2(C)N=N2)C1 c1(NC(c2n(C)cc(NCc3cccn3C)c2)=O)ccc(Br)cc1CC#N C1(C)(C(=O)NCCC(C)(C)NC(c2sccc2F)=O)CCNC1=O CC1CN(C(c2cnn(C)c2C(F)F)=O)CC(C)N(C(C2CSCCS2)=O)C1 Cn1c(O)nc2cc(C(=O)NC3CCCC3NC(C3(C)CCCO3)=O)cnc12 C1(CC(=O)N(C)CCc2cc[nH]n2)CC(NC(c2cc(O)ncn2)=O)C1(C)C N1(CC(N2CCC(CNC(CCC3CCCN(C)C3)=O)C2)=O)CCCNS1(=O)=O C(=O)(C1=CCC(C)CC1)NC1C(CNC(CCc2ncc(C)[nH]2)=O)CC1 c1(C(c2nnnn2C)Nc2c(OC)ccc(O)c2)cc2ccnc(F)c2o1 Cc1nnc(O)c(C(=O)NCC2(C)CCN(C(C3CCOC(C)C3)=O)CC2)c1C N1(C(c2c(CC)nc[nH]2)=O)CC(OC)CC1(C)CNC(c1nnn2c1CCC2)=O CN(CCCC(=O)N1CCN(C(C23CC(N=[N+]=[N-])C2C3)=O)CC1C1CCC1)N=O N1(C(c2cc(F)c[nH]2)=O)CCCC2(CCCN2C(c2cc(F)cc(Br)c2Cl)=O)C1 CC(CC(N)=O)C(=O)N1CCC(NC(=O)COCc2ccnc(O)c2)C(C)C1 n1(CC)ccc(C(=O)NCC2(F)CC(CNC(C3(Cl)CC3(F)F)=O)C2)cc1=O C1(NC(C2(C(=O)NC)CCC2)=O)CC(CNC(=O)CCn2ccnn2)CC1O c1(-n2cnc(NC(N3C(C(=O)OC)CC(OC)C3)=O)n2)nc(Cl)ccc1Cl C#CC1CN(C(=O)CC2(C)CC2)CCN1C(=O)Cc1cncnc1O C1(NS(=O)(=O)CCCCl)CCC(C(F)(F)F)CC1F O=C1C=C2CN(C(C3CCCCN3Cc3ccc(Cl)cc3O)=O)CCC2S1 C(=O)(N=c1[nH]nc(Sc2cccc(C)n2)s1)N(CC(N1CCCC1)C)C c1(C(N(C(C)C(=O)NC2CCCCC2)CC)=O)cnc(O)c(C)c1 c1(NC(C2(F)CN(S(CCOCC)(=O)=O)C2)=O)cc(OC)cc(Br)c1 C=CCC(CC(=O)NCC1(CC(C)C)CCC1)NC(=O)C(F)CCC C(C(CC1CC1)CO)NC(=O)CCN(C(=O)CNC1CC1)CCc1ccccc1 CC1(C)CC2(CC2C(=O)NC2COCCN(C(=O)C(C)(O)C3CC3)C2)C1 N1(C(c2c(OC)nsc2)C(=O)NC2CCCC2)CCCC(Cc2cccnc2)C1 CC(CC(F)(F)F)C(=O)N1CCCC(C)(CNC(c2cnn(C)c2Br)=O)C1 c1(C2C(C)(C)C2)nc(N=c2ccn(C(N3CCOC3=O)C3CCCCC3)[nH]2)cs1 c1(C(N2CCC(N(C(C(CC)=CC)=O)CCC)C2)=O)cnc2cc(OC)ccn12 N1(CCC)CCC(N=c2[nH]c(=NCCCCOCC(F)(F)F)[nH]c3cc[nH]c23)C1 c1(SC(C)(C)C)cc(C(=O)NCCC(O)CNC(=O)Cc2nc[nH]n2)ccn1 C12(NC3C(C)OCC3)CCC(n3cc(CN4CCCCS4(=O)=O)nn3)(CC1)C2 N1(C(Cc2c(C)nc(C)s2)=O)CCC(C)C(NC(c2cnc(N(C)C)nc2)=O)C1 CC#CC1CN(C(=O)CCCN(C)C(C2CC(CC)=NO2)=O)C1 C(C(F)(F)CCC(=O)N1CCC(O)C1C)n1cc(-c2c(OC)cccc2C)nn1 CC(C)C(C(=O)NC1CC(CO)(CO)C1)NC(=O)Cc1nccn1C C(CC(=O)N1CCC(C(N2CCC(N=[N+]=[N-])CC2)=O)O1)N(C)CC Cc1cc(Br)c(C(C(=O)NC2CCC2)N(Cc2ccco2)CC2CCCO2)s1 N1(C(C(CCNC(c2ccc(C#C)cc2)=O)O)=O)CC(C)OC2(CCC2)C1 C=CCC(C(=O)N1CC=CC(NC(=O)CCCCOC)C1)N(C)C N1(C(c2c(O)cc(F)cc2F)=O)CCC2(CCN(C(C3CCOC3)=O)C2)C1 C1(NC(CCN(CCC)C)=O)CCCC(NC(=O)CCOCC(C)(C)C)C1 N1(C(CC2(C(=O)OC)CC2)=O)CCC(C)C(NC(C2CCN(C)C(=O)C2)=O)C1 N1(C(C2CCC(C)(C)C2)=O)CCC2CC1CN(C(c1cnc(OCF)cn1)=O)C2 c1(-n2ccc(C(=O)NCC3C=CCN3C(=O)CSC3CC3)n2)ccc(Cl)cc1 N1(CC(=O)Nc2ccc(OC)c(-c3cc(CO)[nH]n3)c2)CCc2ccccc2C1 C1(NC(C(C2CCOCC2)C)=O)CCN(C(=O)COc2cnc(Cl)cn2)C12CC2 CCC(Cc1ccccc1)C(=O)N(CC(O)CNC(C1(O)CCCC1)=O)C N1(C(C(CC)SC)=O)CCC2(CCN(C(C3(c4cccs4)CC3C)=O)CC2)C1 C=CC1(C(=O)NCC(C)NC(=O)CSc2ccc(C)c(C)c2)CCOCC1 N1(C(CCCSC)=O)CCC(NC(c2cccc(N3CCOC3=O)c2)=O)CC1 CCC(CC(C)C)C(=O)NC(=O)C(C)(C)CF.c12ccc(cc1)C(=O)NOCC2 c1(C(=O)NC(CNC(c2cccc(Cl)c2)=O)C2CC2)cc2ccsc2s1 c1(C(C)OCC)nc(C(=O)NC2(C)CC(NC(=O)CC3OCCCO3)C2)cs1 Cc1nc(C(N2CCCCC2CNC(=O)CC2CC2(Cl)Cl)=O)c(C)n1C1CC1 CC1CCC(C)(C(=O)NCCC(C)(C)NC(=O)Cc2cnccn2)CC1 C(=O)(C(C(=O)NC1CCC(NC(=O)CN(S(C)(=O)=O)C)CC1)OC)OCC c1(OC)ccncc1CC(=O)NC1CCCN(c2ccnn2C)C1 C(=O)(C1COc2cc(F)ccc21)NCC1(C)CCC(C(=O)O)CC1 CC1CN(C(c2cnn(C)n2)=O)CC(C)C1NC(C1CC2C=CC1C21CC1)=O c1(C(C)(C)C)cccc(OCC(N2CCC(NC(C3CCCS3(=O)=O)=O)C2)=O)c1 CP(C)(=O)c1cccnc1NC1CNC(=O)CC12CCC2 CCC(CC)(C(=O)N1CC(CCNC(C2CC(F)(F)CS2)=O)C1)C(C)C c1(C(=O)NC2CC(CNC(CCC(CC)C)=O)C2)c(F)ccc(F)c1OC N1(C(C(F)=CCC)=O)CCN(C(c2cc(C)cc(Cl)n2)=O)C(C(C)C)C1 N1(C(C(c2ccccc2)C)=O)CCOC(CNC(=O)CSCC23CCC(C2)C3)C1 C1(C(N2CCC(OCC=C)CC2)=O)CN(C(=O)Cc2ccnn2C)CC1C1CC1 c1(CN(C(=O)CC(N)Cc2ccccc2)CCCCC)cccc(C#N)c1 N1(C(Cn2c(C(=O)OC)cnc2)=O)CCC(N(C)C(c2sncc2C)=O)C(C)C1 C1(C(N(CCCNC(c2cncc(C(=O)OC)c2)=O)C)=O)CC2CCC1C21CC1 C1(NC(c2c(OC)ccs2)=O)CCC(C(=O)NOC2CCCOC2)CC1 C#CCC(C)(C(=O)N1CC2(CCC2)C1)NC(c1cnsn1)=O C(=O)(C1Cc2ccc(F)cc21)N1CCC2(C(NC(COCC(=C)C)=O)C2)CC1 CC1C(NC(c2cc(Cl)n(C)n2)=O)CCN1C(=O)COCCN(C)C N1(C(C2C(CCOC)C2)=O)CC(O)(CCNC(c2conc2C2CCCO2)=O)C1 N1(C(C(CC=C)C(=C)C)=O)CCOCC2(C1)CN(C(c1ccon1)=O)CCCO2 N1(C(CCc2ccc(C)cc2)=O)CCC(NC(=O)CCC2CCCO2)CC1C C1(NC(C(CCSC)O)=O)CC2CC(C1)N(c1nnc(C)o1)C2 Cc1[nH]c2ccccc2c1CC(N1CCC(NC(C2CCC(=O)N2)=O)C(F)C1)=O C(C1OCc2ccccc21)N(C)Cc1cccn1C1CC1 C1(NC(COCCOCC#C)=O)CCCC(NC(=O)C(C)=C(C)C)C1 CCN=C(NCCCCCC(=O)OC)N1CCC2(CC1)CC2(F)F CC1OC2(CO)CC1(C(N1CCC(C)(CCNC(=O)C(C)CC3CC3)C1)=O)C2 c1(OC)cc(C(=O)NCCNC(=O)C=CCN2CCCC2)cc(OC)n1 C12(C(N(CCNC(C(CC)N(CC)CC)=O)C3CC3)=O)CC3CC(CC(C3)C1)C2 C=CCCCCCCC(=O)N1CCN(C(c2csc(C3CC3)n2)=O)C(C(C)C)C1 C=CCC(F)(F)C(=O)NCC1CC(C(=O)N(C2CC(C)CC(C)C2)C)CO1 C1(O)(NC(=O)COC(F)F)CCN(C(=O)CNC(=O)Nc2cccc(O)c2)C1 N1(C(C(c2cccc(C)c2)=O)=O)C2CCC1CC(O)(CNC(=O)CS(C)(=O)=O)C2 c1(OC)cc(C(=O)N(C2CCCCC2)Cc2ccnc(Br)c2)c(-c2ccsc2)cn1 C1(C(N(CCCNC(=O)Cc2csc(C)c2)CC)=O)CCC2(CCC2)OC1 c1(C(=O)NCC2OCC(CNC(CCCOCC=C)=O)C2)ccc(F)cn1 N1(C(C(n2cc(CCS(N)(=O)=O)nn2)C)=O)CC(C)(C)c2ccc(F)cc21 c1(OC)ccc2c(c1)CN(C(c1cn(C)cn1)C(=O)NC1CC1)CC2 c1(C(=O)NCC(=C)CCNC(=O)CCC2CCCO2)cc(C)c(C(N)=O)cn1 c1(C(N2CCN(C(C(C)C)=O)C(C3CCC3)C2)=O)sc2ncccc2c1Cl Cc1cc(N2CCCC(NC(C3C(C)(C)C3(C)C)=O)C2)nc(C)c1C#N c1(CNC(c2cc(C)oc2C)=O)cc(O)nc(CNC(=O)C(C)OCC(C)C)n1 c1(CNC2CCCC(C(=O)Nc3nc(Br)ccc3Br)C2)c(Br)ccc2c1OCO2 C(=O)(C(CC(F)F)C1CCC1)NCC1N(C(C(=Cc2ccncc2)C)=O)CCC1 c1(SCC)[nH]nc(Cl)c1C(c1nnnn1CCCC1CC1)NC(C)(C)CC n1(CC)cc(CC(=O)N(CCCNC(C2(Br)CC2)=O)C2CC2)c(C)n1 c1(C(=O)NC2CCN(C(c3cc(OC)n[nH]3)=O)CC2O)cc(S(N)(=O)=O)oc1Cl Cc1cccc(CNC(=O)COC2CCN(C(=O)CCCC#N)C2)c1C C#CCCCCC(=O)N1CCCC(CC)C1C(=O)NC(c1cc(C)on1)C N1(C(C(C(C)C)O)=O)CCC(C2(NC(=O)CN3CCP(C)(=O)CC3)CC2)C1 C(=O)(C#CC(C)(C)CNC(=O)C(c1cncn1C)O)NC(CCOC)C c1(C(=O)NCC2CC(c3ccccc3)CO2)cccc2cc(Br)cnc12 CCC(C)C(O)C(=O)N(C)CC1CN(C(c2c(C)nsc2C)=O)CCO1 N1(C(CCCCC=C)=O)CC2(C(=O)NCc3ccc(C)cn3)CCC1CC2 C1(C(N2C(CN(C(=O)CS(N)(=O)=O)C)CCCC2)=O)CC2(C1)CC21CC1 CC1CC(CC(=O)N(CCCN(C(=O)CN2CCN(C)C(=O)C2)C)C)CCC1C C(=O)(C(CC(F)F)N(C(=O)C(CO)NC(N)=O)C)NC1(CNC(C)=O)CC1 CC1(CNC(=O)C=Cc2ccccc2F)CC(F)(F)CN1C(C1CCCCS1)=O C(=O)(C(F)(F)C(O)c1ccccc1)NCC(C)N(C)C(c1cccc(C#N)c1)=O C(CC1CNc2ccccc21)N(C(C(C(C)C1CCCC1)N)=O)Cc1ccccc1 c1(C(C)=O)cc(C(=O)NCC(C(C)(C)C)NC(c2ccoc2C(C)=O)=O)c(C)s1 C1(CC(N2CCC(NC(C3C4CN(C)CC43)=O)C2)=O)CC(C)(C)OC1=O CC1(C(N2CCCC(C(N3CC(N=[N+]=[N-])C3)=O)CC2)=O)CC2(CCC2)C1 C(=O)(C1=CC2CCC(C1)C2)NCCn1cc(C(N(C)Cc2ncc(C)o2)=O)nc1 c1(C(N2CC(NC(C(CC)CC)=O)C(F)(F)C2)=O)cc(Br)c2ccccc2n1 N(C(=NCCC(C)=O)N1CCC(C)(C2CC2)CC1)CC1C(CC)CCCC1 C(=O)(CC(C)C(=O)OC)N1CC(CC=C)(C(=O)Nc2ccccc2N(C)C)C1 C(=O)(C(C)(C)CC1CCOCC1)NC1(C2N(C(C=CCC)=O)CCC2)CC1 C12(OC)CCC(C(=O)NCC(C(C)(C)C)NC(=O)C(C)C(C)C)(CC1)C2 C12(C(=O)NC3(C)CN(C(c4cc5oc(Br)cc5[nH]4)=O)C3)CC1Cc1c[nH]nc12 N1(C(Cc2cn(C)nc2)=O)CCC2(CC1)OCCCC2NC(c1cc[nH]n1)=O c1(C(=O)OC)cnccc1C(=O)NC(C)C(C)NC(=O)C(c1ccccc1)OC CC1CN(C(=O)CCC2CCCCC2)CCC1NC(=O)CCCCN(C)C c1(C(=O)NC2CC(NC(C(C)CC3CCCC3)=O)C2)cccc(N2CCCC2)c1 C1(C(N2CC(C)(NC(=O)C3=CCSC3)C2)=O)CCCCCC(=O)C1 c1(CC)oc2ccccc2c1C(=O)NCC1CC(C)N(C(=O)CN(C)C(N)=O)C1 Cc1nn(C2CCCC2)cc1C(Cc1cccs1)NC(C(C)C)c1cncs1 CC1(C)C2CCC1(C(=O)NC1CCC(CNC(=O)C(Cl)=CCl)CC1)CC2 N1(C(CCCC(C)=O)=O)CC2CN(C(=O)CCc3ccc(Cl)s3)CCC2(CO)C1 N1(C(C2CC(SC)C2)=O)CCC(C)(C(N2CCCC(C(C)C)C2)=O)C1 c1(C(N(C2CN(C(c3c(C(C)C)n[nH]c3)=O)C2)C)=O)sc([N+](=O)[O-])cc1Cl N1(C(C(C)(C)c2cnco2)=O)CCC2CCN(C(=O)Cc3cncs3)C2C1 CCCC(CC)C(=O)NCCn1cc(C(=O)NCC2CCOC(C)(C)C2)nn1 N1(CC(C)NC(C2C3CCCOC23)=O)CCN(C(=O)CCc2cncs2)CC1 C1(CNC(c2c(C)n[nH]c2)=O)CCN(C(=O)CCC(C)(C)N(C)C)C1(C)C C1(CNC(CCSCC)=O)CCN(C(c2coc(C(F)F)n2)=O)CC1(F)F CC1(C)C2CCC1(c1cn(CC(F)(F)CCOC(=N)O)nn1)CC2 CCCC(C)(O)CC(=O)N(C(C)CNC(=O)C(F)(F)CCn1cccn1)C C1(C(N2C(CN(C)C(c3cnn(C)c3Cl)=O)CCC2)=O)CCC(F)(F)C1 C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CCCN(CCNC(C(CC#C)C)=O)CC1 C1(NC(C2CC(OC)C2)=O)CCCN(C(=O)C(O)C(F)F)C1 c1(C(=O)NCC2CN(C(c3c(OC)cc(C)s3)=O)CC2C)cc(F)c(F)cc1O N1(C(C2CCN(CC)C2)=O)CCCN(C(=O)CNC(=O)OC)CC1C C(=O)(C(O)C1=CCCCC1)NC(CNC(c1[nH]cc(CC)c1)=O)CC(F)(F)F C(=O)(C1=COCCC1)NC(CCCNC(=O)CCN1CCC(O)CC1)CO N1(C(=O)OC)CC2(CNC(c3ccccc3-n3cnnn3)=O)CC1CO2 CC(CC(=O)NC1(C)CN(C(=O)C(C)NC(C2CCC2)=O)C1)C1CC1 c1(CC)cc(C)ccn1.C1(C(=O)NCCC2(C(=O)NC)CCC2)CCCN1CC N1(C(CNS(NC)(=O)=O)=O)CC(CO)C2(C1)CN(C(C1CCC=CCC1)=O)C2 C12(CNC(C(C)C(C)(C)C)=O)CCCC(CN(C(=O)C3=CCCC3)C1)C2 N1(C(c2nccc(SC)n2)=O)CC2CCCC(C1)N2C(=O)C(C1CCOCC1)C c1(C(=O)NC2(CCNC(c3n(C)ncc3)=O)CC2)cnn(C)c(=O)c1 CC1(C)CCc2[nH]c(C(=O)NC3CC(O)CN(C(=O)CCC(N)=O)C3)cc2C1 C1(N(C(C(C)=C(C)C)=O)C)CCC(NC(=O)CCn2cccnc2=O)CC1 C(C1CN(C(c2cc(C3CC3)no2)=O)Cc2ccccc21)NC(C(C=C)(C)C)=O C=CCCCC(C(=O)N1CCC1C(C)O)NC(=O)Cc1ccco1 C1(O)(CCNC(c2c(C(C)(C)C)c[nH]c2)=O)CCN(C(c2ccc(O)nn2)=O)C1 C1(C)(CNC(c2c(C)nc(C)o2)=O)CN(C(=O)COCCN(C)C)CC1C c1(NC(C)=O)ccc(C(N2CCC(NC(C3CC(=O)N(C)C3)=O)C2C)=O)nc1 C1(CC)(NC(c2ccccc2OC)=O)CCN(C(c2cc(OC)n(C)n2)=O)CC1 C(=O)(CC(C)(C)C#N)N1CCC(C(C)NC(c2csc(CC3CC3)n2)=O)C1 C1(C(=O)NC(c2ccc(C)s2)C)CNC(=O)CN1C(C1CC2CC(=O)C1C2)=O Cc1cc(=NC(=O)CN2CC(NC(=O)C(C)OCc3ccncc3)C(C)C2)[nH]o1 N1(C(C2C(C)OCC2)=O)CC2CCCN(C(=O)COc3ccc(Cl)cc3Cl)C2C1 c1(OC)cc(N)c(C(N2CC3(C2)CN(C(c2cc4c(s2)CCC4)=O)C3)=O)cc1F c1(C(=O)NC2(C)CN(C(C(C)Cc3ccncc3)=O)C2)cc2cc(Cl)ccn2n1 N1(C(Cc2cncc(C)c2)=O)CCC(NC(=O)CSCC(N)=O)CC(O)C1 C1(C(=O)Nc2c(OC)ccnc2)CCC(C)N(C(C2COCC(C)O2)=O)C1 c1(CNC(C=C)=O)ccccc1S(=O)(=O)CC(CN(C)CCC)OC c1(-c2cc(C(N3CCCC3)=O)no2)ccccc1F.N12CC3C(C3C1)NC2=O C1(CC(=O)N(C2CCN(C(c3cc(C4CCCC4)[nH]n3)=O)C2)C)CCC(C)(C)C1 c1(C(N(C2C(CC)CCC2)C)=O)ccnc(C)c1O c1(CC(=O)NC2COCCN(C(c3c(C)nc(C)o3)=O)C2)c(F)ccc(F)c1F Cc1cccc(CC(=O)N(CCC(C)NC(=O)C(F)n2cccn2)C)c1 c1(OCC)cccc(C=CC(=O)NC(CNC(c2snc(Cl)c2Cl)=O)CC)c1 N1(CC(=O)NC2(CNC(=O)Cc3nc[nH]c3Br)CCC2)C(=O)CCC1=O CN1N=CC(CC(=O)NCC(C)(C)CCNC(C2CC2F)=O)C1=O n1(CC(C)C)[nH]c(CC(=O)NC2(CNC(=O)C(F)C3CCC3)CC2)cc1=O c1(C(=O)NCC(O)CN(C)C(C2(CC)CC2(F)F)=O)cc(CO)n(C)n1 c1(C(N(C)CC2(NC(C(C)NC(C3CCCC3)=O)=O)CC2)=O)ccc(Br)o1 C(=O)(CC(C)(C)COC(C)=O)N1CCC(NC(COC)=O)C1c1ccccc1 C1(C(=O)NC2CC(CC(=O)NC(C)C(=O)N(C)C)C2)CCCN1C(N)=O c1(C(C(=O)NCC(F)F)N(CC(=C)C)CCOC)cc2cc(Cl)ncc2o1 N1(C(CCC=C)=O)CC(C2CCN(C(=O)CCC(=O)OCC)C2)C1 C1(O)(C(N2CC(C)N(C(c3cnc(S)n3C)=O)CC2)=O)CCCC(C)(C)C1 c1(OC)ccc(CO)cc1C(N1CC(NC(c2coc(C(F)F)c2)=O)C(O)C1)=O C1(CC(=O)N(CCN(C(C(C)NC(CC)=O)=O)C)C)COC(C)(C)CO1 c1(CN2CCC(CNC(c3ccc(NC)cc3)=O)C(C)C2)c(C)cc(Cl)cc1Cl c1(C(N2CCC(CNC(C3=C(C)OCCS3)=O)CC2)=O)c(C)nn2c1CCCC2 C1(C(N2CC3C(NC(C4CC(OC)C4)=O)C3C2)=O)CCCCC1(F)F c1(C(N2C(COC)CN(C(=O)C(=O)N(C)C)CC2)=O)cc(C)c(O)c(C)c1 C12(NC(COCC)=O)CCC(CC1)N(C(c1cc3nccnc3[nH]1)=O)C2 C=C(C)C1OCCCC1C(=O)N(CCNC(=O)C(C)(C)NC(=O)C(F)(F)F)CC N1(c2c(C)c(NC3CCN(CC4CC4)C3)ncn2)CCCC2(CCN(C)C2)C1 C1(NC(C(C)CN(C)C)=O)CN(C(=O)CC(F)(F)Cl)CC12CCCC2 C1(NC(=O)NC2C(C)(CC)C2)CCCOC1(C)C CCC(C)C(C)CNC(C1CCN(S(=O)(=O)Cc2ccccc2OC)CC1)=O CC1CN(C(=O)CCc2cscc2Br)CCC1NC(c1nccnc1N)=O c1(C(N2CC3C(NC(C(C=C)CC)=O)(C3)C2)=O)ncnc(C)c1C c1(CC)c(C(=O)NC(CNC(C2(O)CC2(C)C)=O)C2CC2)nnn1CC c1(CN(CC(C)C)C(=O)NC(c2ccc(OCC)cc2)C)nccc(C)c1F C(=O)(CC(=O)NCCN(C)C(c1cc[nH]c1)=O)OCCC(C)C c1(OC)cc(C(=O)N(CC(O)CN(C)C(C2C3CCCCC23)=O)C)c(Cl)cn1 C(C(C)(CC)C(N)=O)NC(C(CNC(C(C(C)OC)N(C)C)=O)OC)=O C1(NC(C=CSC)=O)CN(C(C2CCC(=O)N(C)C2)=O)CC12CCOCC2 Cc1cnc(C(=O)NCc2ccc(C3CCCCC3)o2)nc1 N1(C(C(C)OCC(C)C)=O)CCC2(CCCCC2NC(=O)CC2CCCCO2)C1 c1(C(=O)NCC=C=C)cc(C(=O)NCC2CCCN(CC)C2)nn1C CC(CC(=O)N1CC2CCCC1C2CNC(c1coc(C(N)=O)c1)=O)C(C)(C)C C1(C(=O)OC)COCC(C)N1c1ccc(C#N)cn1 c1(C2C(C(=O)NCC(C)(O)CNC(=O)C(O)c3ccco3)C2)ccccc1Cl Cc1ocnc1CC(=O)NC1(CCC(=O)NCC(C)(C)C2(O)CCC2)CCCC1 c1(CC(=O)NCC(=C2CN(C(C(C)OC3CCCC3)=O)C2)F)ccccc1CO N1(C(C(CCSC)NC(c2ccccc2)=O)=O)CCOC(C)(CNC(=O)CO)C1 N1(C(CC2CC(C)C2)=O)CC2(CCC(CNC(c3cc(C(F)F)n(C)n3)=O)O2)C1 C1(C(N(C2CCN(C(=O)CCOCCN(C)C)C2)CC)=O)CCCC1(F)F CCC(C)CCC(=O)NC1CCN(C(C2CC2c2cncs2)=O)CC1 N1(C(C2CC(=O)N2)=O)CC2CCCC1C2CNC(=O)C(F)=C1CCCC1 c1(CC(=O)NCCN(CCC)CCOc2ccccc2)ccc(O)cn1 C1(C(C)CNC(=O)C(c2cccnc2)C)CCN(C(=O)C2=NOCC2)CC1 c1(C(C)(C)C)ncsc1C(=O)NCC1CC1CNC(=O)Cc1n[nH]c(=N)s1 C1(C(=O)NC2(CC=C)CN(C(=O)C(C)(C)C(N)=O)C2)CCC(C)(C)CC1CN O=C(N=c1nc[nH]n2cccc12)C1CC(F)CN(C(=O)C2=CCCCO2)C1 c1(-c2cn(C3CN(C(C(C)OC)=O)CC3C)nn2)ccnc2ccccc12 CC(C)C(C(=O)NCCc1cccc(O)c1)NC(c1nnsc1N)=O N1(C(C(C#C)(C)C)=O)CCC(C(=O)N(C2COCC2OC)C)CC1(C)C N1(C(C(CC(C)C)O)=O)CCC2OCCN(C(=O)CCc3ccccn3)C2C1 C12(NC(c3cccc(-n4cc(-c5cscn5)nn4)c3)=O)CCC(CC1)C2 N1(C(Cc2ccc(OC)cc2C#N)=O)CCC2(CCC(C)C2)C1 C(=O)(C(C)CC(C)C)NCCCNC(c1c(CC)occ1)=O c1(N)ncc(F)cn1.C1(NC(C2CC2C(F)F)=O)(C)CCC1.C12(CC1)C(=O)NC2 O(NC(=O)C1=CC2(CN(C(=O)C(C)CC=C)C2)OC1)CCC#C c1(C(N(CCCNC(=O)COC2CCOC2)C(C)C)=O)cc2n(n1)CCCO2 C(=O)(C#CC(C)(C)O)NC1C(N2CCN(C(C3(CC=C)CC3)=O)CC2)COC1 n1(CCC(=O)NCC23CCC2CN(C(c2cccnn2)=O)C3)ccc(O)nc1=O c1(C(=O)NC2(COC)CN(C(C3CC4(CC4)C3)=O)C2)cc(F)cc(N)c1F CCC(CC(=O)N1CCN(C(=O)Cc2sc(C)nc2C)CC(O)C1)C(C)C N1(C(C2C(CC)OCC2)=O)CC=C(CNC(c2csc(C(C)C)n2)=O)CC1 C=C(C)C1OCCC1CNC(=O)NC(C(=O)N(C)C)C(C)(C)C c1(C(N2CC(C)(NC(Cc3nc(C(C)C)sc3)=O)C2)=O)ccc([N+](=O)[O-])o1 CC1(CNC(=O)C(C)(C)CCF)CCN(C(c2cc(C(C)(C)C)c[nH]2)=O)CC1 CC(C)(CCCNC(=O)C(C)(C)n1ccc(C2CC2)n1)NC(C1CC=CC1)=O c1(C(=O)OCC)noc(CNC(=O)C(c2ccccn2)N(C)C)n1 C1(CNC(C2(CO)CC(C)(C)C2)=O)CC(C(=O)N2CC3(C2)CC3(F)F)=NO1 CC1CN(C(C23COCC(C2)C3)=O)CC(C)C1NC(c1cnc(C2CC2)s1)=O c1(C(=O)NCc2ccc(CNC(=O)CC3CCC3)cc2)c[nH]c2ccc(O)cc12 c1(CN2CC3C(NC(c4nn(CC)c(C)c4)=O)C3C2)cc([N+](=O)[O-])cs1 C#Cc1cnc(NC2CCC(CNC(=O)CSc3ccccc3)CC2)nc1 c1(-c2cn(CCC3CC(NC(c4c(Br)n[nH]c4Br)=O)C3)nn2)ccc(Cl)c(Cl)c1 c1(C(=O)NC(CC)CNC(=O)C(C)CC)ncc(C)cn1 C1(CC)COCC1NC(=O)C(CC1CCOCC1)NC(C1(c2cc[nH]n2)CC1)=O C(=O)(CCC(C)(C)F)NCCC(C)NC(CCc1cc(OC)no1)=O Cc1nc(C(C)C)ccc1C(=O)NCC1CC2CN(C(=O)C(C)(C)C(F)F)CC12 C1(NC(C2CCC2)=O)CCCC12CN(C(c1cc(C3CC3)oc1C1CC1)=O)C2 Cc1cc(C)nc(CC(=O)NC(C2CCN(C(=O)C(C)NC=O)CC2O)=O)n1 C(N=c1nc(N2CCOCC(CO)C2)c2ncn(C)c2[nH]1)C1N(C)CCOC1 c1(NC(=O)C(c2ccc(F)cc2)O)ccc(-c2cccnc2)cc1 C1(CC(C)O)CCCCN1C(=O)C=CCN(C)C(c1cnn(C)c1)=O c1(CC(N2CCC(NC(c3c(C)cno3)=O)C(C)C2)=O)ccc(C#N)cc1F CCC(CNC(=O)CC1CCCCN1C(=O)CN1CCCNC1=O)CCO C1(CCC(=O)NC(CNC(c2ccc(O)cn2)=O)CO)CCC(O)CC1 C1(C(N2CCC(CNCc3ccn(CCF)n3)CC2)=O)CCCCC1(F)F Cc1nc(NC(C)CCC(C)(C)C)cc(=NC(C)c2cc(C(F)(F)F)nn2C)[nH]1 N(C1CCCn2nccc21)c1c(C(=O)NCC2CCCO2)cccn1 c1(C(N(C2CN(C(c3cccc(I)c3Cl)=O)C2)C)=O)nccc2nc[nH]c12 C1(NC(c2c(OC)ccs2)=O)CCCN(C(=O)C(F)CC(C)C)C1C C1(=O)C(C)(C)Cc2cn(nn2)C2COCC12.n1(CC)ncnc1C(=O)NC1CC1 C1(NC(C(C)OCOC)=O)CC2(CCCCN2C(c2cnc3[nH]ccc3n2)=O)C1 N1(C(Cc2ccn(CC)n2)=O)CCN(C(=O)CC2CC(C(F)F)C2)C(CO)C1 N1(C(c2cc(C)no2)=O)CCC(NC(=O)C(c2ccc(Cl)cc2)C)C1(C)C Cc1cc(C(=O)NC2CC(NC(c3cncn3C)=O)C23CCC3)c(C)n1C C1(CNC(c2cc(C(C)C)[nH]n2)=O)CCC(CNC(C2CCCCO2)=O)CC1 Cc1c(CC(=O)NC2CN(C(C3(F)CC=CCC3)=O)CC2O)cccc1[N+](=O)[O-] C1(CCC)CN(C(C2CCCN2C(=O)N(C)C)=O)CCN1C(=O)CCCF S(=O)(=O)(c1ccc(C(N2CC3CNCC3C2)=O)cc1)NC(C1CCCC1)C C(c1ccncc1)=CC(=O)NCC(c1ccccc1)NC(C1CCCS1)=O C(N=c1nc2c(cnn2C)c(NC2CC3CCC(C2)C3O)[nH]1)C1(C=C)CCC1 CC(CC(=O)N1CC2(CC(CC(=O)NC(CCO)C3CCC3)C2)C1)C(F)F c1(N(CC(C)C(F)(F)F)C)cccc(S(=O)(=O)NCc2sc(Cl)cc2Cl)n1 C(=O)(CCS(C)=O)NCC1C(NC(c2ccc(COC)s2)=O)CC1 n1(CC(=O)NC2(O)COC2)cc(COC2CCN(S(=O)(=O)CCC)C2)nn1 c1(C(=O)NCCOC2CN(C(c3cn(C(C)C)nn3)=O)C2)cccc(=O)n1C C(=O)(C1=COCCO1)NC(C1CCCCC1)CNC(c1ccc(OC)s1)=O C1(NC(c2ccc(SCC)nc2)=O)CN(C(C2CNC(=O)N2)=O)C2CCCCC12 O=C1CCC(CCC(N2CC3C(NC(C4(C5CCC5)CC4)=O)C3C2)=O)CN1 c1(N2CCN(C(C(C)OC)=O)CC2)ncnc(N2CC3CC2CO3)c1C c1(C(N2CC3C(CN(C)C(c4csc(CO)n4)=O)C3C2)=O)ncc(C#N)cc1Cl C1(C(N(CCN(C(C)C)C(c2cnc(S)nc2)=O)C)=O)CCCC(=O)CC1 S(=O)(=O)(c1cccnc1NCc1ncsc1C)NC(c1ccccc1Cl)CC Cc1nc(C)c(C(=O)NC23CC(NC(C4CCN(C=O)C4)=O)(C2)C3)s1.C1(CO)CC1 C1(C)(C(=O)NC(C)C(C)(C)NC(C2CC(=O)N(CCN(C)C)C2)=O)CC2(CC2)C1 Cn1c(C(N2CCCC(CNC(C3Cc4nnsc4S3)=O)C2)=O)cccc1=O N1(C(C(c2cc(F)cc(F)c2)=O)=O)CCCC2(CCN(C(C3(O)CC3)=O)C2)C1 CN1CCOc2ccc(C(=O)N(C)CC3CCCN(C(c4ccon4)=O)C3)cc21 C(C)(C(=O)N(C(C)C)CC1CCC1)N(C(CNC(C)=O)=O)C c1(C(=O)NCC2C3CN(C(C(CC)=CCCC)=O)CC32)cc2sc(C)nc2[nH]1 c1(CC(=O)NC(C)CC2CN(C(C3OCC3(C)C)=O)C2)ccc(F)c(Cl)c1F c1(C(=O)NC(CN(C(=O)C(C)C(C)(C)C)CC)C)ccc(Cl)c(F)c1N N1(C(C(C)CO)=O)CC(NC(c2ccc(P(C)(C)=O)cc2)=O)Cc2ccccc21 c1(N2C(C(=O)NCC3CCC3)C(O)CC2)ncnc2ccc(I)cc12 Cc1cc2cc(C(=O)NCC3CC3CNC(=O)C(C)C3CCOC3)ccc2cn1 N1(C(C(C)NC(c2ccoc2)=O)=O)CC2CC3CC2C1C3NC(=O)C1=CCC1 c1(CC)cc(C)c(C(=O)N(C)CC2CN(C(=O)Cc3sc(S)nc3C)CCO2)o1 C1(C(=O)NC(c2ccc(N(C)C)cc2)C)CCC(F)CN1 n1(CC)cc(CC(N2CC(N(C(=O)CNc3ccccn3)C)C2)=O)cn1 N1(C(C=CC)=O)CCCC2(CCN(C(c3ccc(NS(C)(=O)=O)cc3)=O)C2)C1 c1(C(=O)NCCC2OCCN(C(C(C)CF)=O)C2)cc(Cl)cc2ccccc12 N1(C(c2c(OC)cc(C)cn2)=O)CC(NC(=O)C(C2CC2)SC)CC12CCC2 C1(NC(CCN(CCC)C)=O)CCCCCC1NC(=O)C(C(C)C)SC O=C1CC2CCCC2(C(N2CCOC(CNC(c3cc(C(F)F)[nH]n3)=O)C2)=O)C1 c1(C(=O)Nc2cccc(-c3cn(CCC(=O)OC)nn3)c2)c(Cl)cc(Br)cc1Cl C1(NC(c2cc(C)oc2)=O)COC2(C1)CN(C(=O)C(O)CC1CC1)C2 C1(C(=O)NCC2(NC(c3ccc(N)c(N)n3)=O)CCC2)COc2ccccc2O1 n1(COCC)nnc(C(=O)NC(C)CNC(=O)CC(c2cccc(F)c2)O)c1N c1(C(=O)NC2(CCNC(C3CCCC(C(N)=O)C3)=O)CCC2)ccnc(Cl)c1N N1(C(C(=Cc2cccnc2)C)=O)CCC2(CCCC2NC(=O)Cn2ccnn2)C1 C(C(COC)CC(=O)N1CCOC(C2CC(NC(=O)CCCOC(C)=O)C2)C1)OC N1(C(c2nccs2)C)CCN(c2ccc(C(F)F)cn2)CC1 CN1CCCC(OC(=O)C=Cc2cncn2C)C1=O c1(CNC(C2(c3ccc(-c4cnc(C)s4)cc3)CCCC2)=O)cccc(Br)c1O C1(NC(C2CCN(C(=O)CN3CC4CC4C3)CCO2)=O)CCCC(C2CC2)C1 C(=O)(CCC(C)(C)c1ccccc1)NCC(C(C)C)NC(=O)CC12CC(C1)C2 N1(C(c2nc3cccnc3s2)=O)CC2CCCC(C1)N2C(=O)CSc1cccs1 CC(C)CS(=O)(=O)CC(=O)NCC1(F)COCCN(C(=O)COC2CCC2)C1 c1(C(N(C)CC2N(C(Cc3cc(C)ns3)=O)CCOC2)=O)cnn2ccccc12 C(CCCCC(=O)NC1CC1CNC(c1ccc(F)c(Cl)c1)=O)NC(N)=O CC1(C)CN(C(=O)CCP(C)(C)=O)CC1CNC(C1CCS(=O)(=O)C1)=O C1(C#CC(=O)N2CC3(CC(CNC(=O)C=C(C)C)C3)C2)(CC)COC1 c1(CCC(=O)NCCCCNC(C2CSCCS2)=O)cccc(F)c1 C1(CC(=O)N(C2CCN(C(=O)CC(C)(C)C)C2)C)CCCC(=O)N1 C1(C(N2CC3CC2CO3)=O)CC(F)(F)CN1C(c1cccc(Br)c1Cl)=O C1(NC(c2cncc(COC)c2)=O)COCCN(C(C2(O)CCCCC2)=O)C1 C1(NC(C(C)(C)c2ccccc2)=O)CCCC(NC(c2cc(C#N)c[nH]2)=O)C1 C1(C(=O)NC2C3(CC(NC(CCCC=C)=O)C3)C2)CCCCC1N=[N+]=[N-] C1(CC=C)(NC(C2CC(=O)NC(C)C2)=O)CCCN(C(=O)C(C)=C(C)C)C1 C(C(C)(C)CNC(=O)CCC1CCOCC1)N(C(c1c[nH]cc1C)=O)CC c1(C(=O)NCC2CC(CNC(COCCC)=O)OC2)ccc(C2CC2)cc1F C1(C(N(C)CC2CCN(C(=O)C=CC3CCCO3)C2)=O)C2CC3C(C2=O)C13 C(C(CNC(C1CCC1OC)=O)C(F)(F)F)NC(c1c(CC)onc1)=O C1(NC(C2N(C(C(C)=C3CC3)=O)C3(CC2)CC3)=O)CCN(C)CC1C#N C1(NC(COC2(C)CN(C(c3cc(C)sc3C)=O)C2)=O)CCCCC1C#N CN1CCN(C(C2C(F)(F)C23CCC3)=O)C(CNC(=O)CCc2nccs2)C1 C1(NC(=O)Cn2nccn2)CCCN(C(=O)CSCc2ccccc2)CC1F N1(C(CC2C(C)=NOC2=O)=O)CCCC(C2(NC(=O)CC3CCSCC3)CC2)C1 C#Cc1ccc(Cl)c(C(=O)NCCOC2CN(C(C3(O)CCSC3)=O)C2)c1 c1(CN(C(N2C(CN=[N+]=[N-])CCC2)=O)C2CC2)nc(C)c(C)o1 CC#CCCCC(=O)N1CCN(C(=O)C(O)CSC)C(c2nccn2C)C1 C12(CNC(=O)NC(C(CC)CCO)C)CCCCC(=O)N1CCC2 N1(C(C2(CC)CC2)=O)CCC2(CC1)CC2CNC(=O)CC1CNC(=O)C1 C1(C(N2CC(C(C)(C)C#N)C2)=O)N(C(C2CCC(=O)CC2)=O)CCC1(C)C c1(CC)cc(F)c(C(=O)NCCC(C)NC(c2n[nH]c3c2COCC3)=O)cc1F N1(C(C(C)C2(O)CCC2)=O)C(C(=O)NCCCc2cc[nH]n2)CCC12CC2 C1(CCCC)CN(C(=O)C(=O)NC2CC2)CCN1C(=O)CCc1ccccc1C C12(NC(Cc3nnc(C)n3C)=O)CCC(CC1n1cc(CCS(C)(=O)=O)nn1)C2 c1(OC)cc(OC)c(C(=O)NC(CNC(=O)CNC(N)=O)C(C)C)cn1 CC1CCN(C(=O)CCCc2nccs2)CC1NC(c1scnc1C1CC1)=O C#CCCCCCCC(=O)NCC(CC)NC(=O)Cc1c(C)n[nH]c1C c1(CC(=O)NCCC2(C(N(C3CC(C)C3)C)=O)CCC2)ccc2occc2c1 C1(CC(=O)NC2CCCCN(C(=O)C=Cc3cncs3)C2)CCC2(CC1)CC2 N1(C(CC2CC(=O)NC(=O)C2)=O)CC2CCN(C(C3CSC(=O)N3)=O)C2C1 c1(NC(C2(N(C(=O)CC3CC(F)C3)C)CC2)=O)ncccc1Cl N1(C(C2CN(S(CC)(=O)=O)C2)=O)CCCC(O)(CNC(=O)CCP(C)(C)=O)C1 CON(CC1CC2CCC1C2)C(=O)Nc1ccccc1-c1nc(S)n[nH]1 c1(CC(=O)NC(C2CCN(C(c3cnc(OC)s3)=O)C2)C)cc(O)nc(O)n1 c1(C(=O)NC2(CC=C)CCN(C(C3CCCCC3C)=O)C2)cccc2[nH]ncc12 Cc1cncc(CNC(=O)C(C)CC2CCCO2)c1 C1(CNC(C(c2cccc(Br)c2)C)=O)CCN(C(c2ncccn2)=O)C1(C)C Cn1nc(C2CC2)cc1CC(N1CC(NC(=O)CC2(C)CCCCC2)C2CC12)=O N1(C(c2cc(C(C)(C)C)no2)C(=O)NCCC(=O)OCC)CCN(C)C(C)C1 Cc1ccc(O)c(NC(=O)CC2CN(C(=O)CCc3cn[nH]c3)CC2C)c1 S(=O)(=O)(c1ccc(C(=O)OCc2cc(C#N)ccc2C)cc1)N(CCC)C N1(C(C(N)=O)=O)CCC2(CC2C(=O)Nc2cc(Cl)cnc2O)C1 CC1CN(C(=O)CCCc2ccsc2)CCCN1C(=O)COC1CCCC1 Cc1cc(C)n(C(C)CNC(=O)N(O)Cc2cn(C)cn2)n1 N1(CCNC(c2ccc(COC)o2)=O)CCN(C(=O)C(O)c2ccco2)CC1 c1(C2(C)CC2C(=O)NC2CC3CN(C(C4CN(C)C4)=O)CC23)ccc(F)cc1F N1(C(C(C)S(N)(=O)=O)=O)CCC2(CCCC2CNc2cc3nncn3cn2)CC1 c1(NC(C)=O)ccc(F)c(C(N2CC(C)(NC(c3csc(C#N)c3)=O)C2)=O)c1 CCC(C)CC(=O)C(=O)N(C1CN(C(=O)CCn2cc(C)cn2)C1)C S(=O)(=O)(CC(=O)NC1(CNC(C2CC2C(C)(C)O)=O)CCC1)N(C)C O=C(C1=CCC2(COC2)OC1)NCc1nccc2occc12.C12CCN1C2=O C(=O)(CC(C(C)OC)NC(c1ccc(C(C)=O)o1)=O)NCCC(CC)(C)C N1(C(C(C)C2CCOC2)=O)CCC2(CCCN2C(=O)Cc2csnn2)C1 c1(C(=O)NC2C(NC(c3cc(CC)on3)=O)CCC2)cnn(C)c1-n1cccc1 CCCC(CCC)C(=O)N1CCC(CCC(N2CCC(O)C(CC)C2)=O)C1 CC1CSCCN1C(C1CCCC(NC(=O)C(=O)NCC(F)F)C1)=O c1(C(N2CC(C3CN(C(C(CC)(C)CO)=O)C3)C2)=O)cn2cc(C)sc2n1 c1(C(N(CCCCNC(C(C)SC)=O)C)=O)cccc(C#N)c1Br c1(CC(=O)NCCCNC(C=CCCC)=O)csc(-c2ccccn2)n1 c1(CC(C(=O)NC2CCOC2=O)NC(C2CCSCC2)=O)ccccc1Br C(=O)(CS(C)(=O)=O)N(C)CC1(O)CN(C(C(N2CCOCC2=O)C)=O)C1 C1(NC(c2n(C)nc(CNC(=O)CC3(C#N)CC3)c2)=O)CC(O)CC(C)(C)C1 c1(C(=O)NCC2(F)CCN(C(c3c(CC)n(C)nn3)=O)C2)c(OC)ncnc1C C1(CCC=C)(C(=O)Nc2cc(C(N)=O)no2)CN(C(=O)COC2CCCC2)C1 C1(CNC(C2(OC)CCN(C(=O)C(=O)OC(C)=O)C2)=O)C2CCCCCC12 C(CCCCC(=O)N(C1C2CN(C(c3c(C)nsc3N)=O)CC12)C)NC(C)=O c1(C(=O)NCC2OCCN(C(C3(C=C)CC3)=O)C2)cnc2ccnn2c1C c12ccc(C(=O)CN3CC(OC)C3)cc1C(=O)CCOCC(=O)NC2.CCN C1(NC(c2c(Cl)ccc(C)c2)=O)CC2CCC1CN2C(c1cnnn1C)=O CCC(O)C(C)(C)C(=O)N1CCCCC(N(C)C(c2ccnc(C)c2C)=O)C1 N1(C(c2ccncn2)=O)CCC2CCCC(C1)N2C(c1cnc(Cl)s1)=O c1(CC(=O)NC2CCC(CS(=O)(=O)Oc3ccccc3F)C2)ccccc1F c1(C(=O)NCCN2CCN(C(c3nn[nH]c3Cl)=O)CC2)ccc2nc(O)[nH]c2c1 C1(C(=O)NCC(N(C)C(c2cn(CCCF)nn2)=O)C2CC2)CCCCC1(C)C N1(C(C(C)c2ccco2)=O)CC(NC(=O)Cc2csc(Br)n2)CC2(CC2)C1 Cc1nc2cccc(C(=O)N(C3CN(C(c4cc5nc(C)sc5[nH]4)=O)C3)C)c2[nH]1 C1(NC(c2ccc([N+](=O)[O-])nc2)=O)C2CCC1CN(C(C1(F)CCCCC1)=O)C2 N1(CC)CCN(C(=O)CC(C)CNC(c2nc(C)ccc2F)=O)C(C)C1 c1(C(=O)NC(CC)C(=O)NC(C2CCC2)C)cc(O)cc(F)c1 c1(CN(C(=O)CCN(C2CC2)C(C2CC=CCO2)=O)C)cccnc1O N1(C(C(C)OCCC=C)=O)C(CNC(c2ccn(C)c(=O)c2)=O)CC2CCCC12 c1(C(N2CCC(NC(C(C)Cc3ccco3)=O)(CF)C2)=O)nc(O)nc(O)c1N C12(C(=O)NCC(n3c(C)ncc3)C)CC(C1)C(C)O2 c1(C(=O)NC2C(NC(c3ccc(C#N)cc3)=O)CCCC2)ccc2n[nH]cc2c1 N1(C(C23N(C(CN(CCCCCC)C)=O)CC(C2)C3)=O)CCc2c[nH]nc2C1 c1(C(=O)NCC(C)(C)NC(Cc2n(C)c(C(F)(F)F)cn2)=O)ccc(F)cc1O C=C1CCC(C(=O)NOCC(=O)NCC2CC(CCO)C2)CC1 C(=O)(CC(COC)COC)N1CC(CC)C(C(=O)Nc2ccc(C)cc2C)C1 C(=O)(N=c1cnn(C)[nH]1)C1CCC(NS(CC=C)(=O)=O)CC1 c1(C(=O)NCC2C(CNC(CCOC(C)C)=O)C2)cccc2cncn12 C1(NC(CCC#CC)=O)CC(C)CN(C(=O)CC2(C(F)(F)F)SCCS2)C1 CCC(CN1CCCC1)N=c1ccnc(N2CCC(F)(c3ccccn3)CC2)[nH]1 C1(C)(CNC(c2nc(C)sc2C)=O)CN(C(=O)CC2(N3CCCC3)CC2)CCO1 C1(C(=O)NCc2n(C)nc(C(F)F)n2)CC2C=CC1C21CC1 c1(CC(=O)OC(=O)C(O)c2ccco2)ccc(F)cc1.CC1C(=O)N(C)C1=O C#CC1(C)CCN(C(=O)CC2C(NC(C3(C#C)CC3)=O)CC2O)CC1 C1(C(=O)NCC(=O)Nc2ccccc2)C2CC1CN(C(C1CC13CCOC3)=O)C2 c1(N2C(C)CC(NC(c3c(CCC)nco3)=O)C2)cc(C)c([N+](=O)[O-])cc1F C1(NC(c2cc(Br)n[nH]2)=O)CCCCC1C(=O)NCC1CC(N2CCCC2)C1 CC1CN(C(=O)NCc2nn[nH]c2C(F)(F)F)CC1CCc1ccccc1 c1(C(=O)NC)cccc(CCC(=O)NC2CN(C(C3CC(Cl)(Cl)C3)=O)CC2C)c1 C1(OCC)CCN(C(=O)C=CCN(C)C(C2CCN(OC)CC2)=O)CC1C c1(OC)nc(C)ncc1C(=O)N(CCN(C)C(C1CN(C)C(=O)N1)=O)C(C)C C1(NC(CCn2ncc(C)c2)=O)CC2CC1N(C(c1nc(O)c(C)s1)=O)C2 c1(CNC2CC(NC(C(c3ccccc3)SC)=O)C2)cccc(C(C)(C)C)c1 c1(OC)ccc(N2CCCC2c2ccccc2I)cc1-c1cccnc1C#N c1(-c2nnc(N(C(c3cccnc3)C)C)n2C)cnc2c(c1)COC2 CC(CN(C)C(c1cc(CNC(=O)C(O)c2ccsc2)no1)=O)C(C)(C)C c1(CC(=O)CCN(C(=O)CC2CCC(=O)N2)C)cccc(OC(F)F)c1 N1(C(C2CCN(C(=O)NC)CC2)=O)C2CCC1C(C)C(NC(C1(O)CCC1)=O)C2 CN1CC(NC(C2(NC(C3CCCO3)=O)CCC2)=O)CC1=O c1(N2CCCC(C)(NC(c3n[nH]c(C)c3C)=O)C2)ccc([N+](=O)[O-])cc1Br c1(C(=O)NC(C2CN(C(CC(CC)(F)F)=O)C2)C)ccc2c(c1)C(C)C(C)O2 CC1=C(C(=O)N(CC(=O)NC2CCCN(O)C2=O)C2CC2)COCC1 Cn1cc(C(N2CCN(C(=O)C(F)C3CCC3)CC2CO)=O)c2ccccc12 N1(C(c2cnc(SC)s2)=O)CC2(C1)CN(C(=O)CCN1CCCC1=O)CC2CO CC(CC(=O)N1CCC(C)(NC(=O)C(=O)C=Cc2cccs2)CC1)CC(C)(C)C C1(C(=O)NC2(CC=C)CN(C(c3[nH]nnc3C)=O)C2)C(Cl)(Cl)C12CC2 Cc1cccc2nc(C(N3CCCC(O)(CN(C)C(c4cnn[nH]4)=O)C3)=O)cn12 CC(Cc1cccnc1)C(=O)NC1(CF)CN(C(=O)C(C)CN2CCOCC2)C1 N1(C(Cc2c(CC)con2)=O)CC2(COC(CNC(=O)CN(C)CC)C2)C1 N1(C(C(CCCC)=O)=O)CCN(C(c2cc(=O)cc[nH]2)=O)CC(C)(F)C1 C1(NC(c2ccc(C)cc2)=O)CCC(C)N(C(C23CC(NC(=O)OC)(C2)C3)=O)C1 C(=O)(CC(C)C(=O)NC(C1CCCCC1)CNC(=O)Cc1ccc(O)cc1)OC N1(C(c2c(NC)cncc2)=O)CCCC12CCN(C(=O)C(c1cnccn1)C)C2 N1(C(CC(C)n2cccc2)=O)CC2CC(NC(=O)C=Cc3cscn3)C1C2 c1(C(N2CCC(C(=O)NC3COCC3CO)(OC)C2)=O)nc(C)ccc1F c1(C(N2C(CN(C(C(C)OCC)=O)C3CC3)CCC2)=O)cc(O)n(C)n1 O(N1CCC(CC(=O)NCC(CC)NC(=O)C(O)CCSC)CC1)CC C1(CN)(CO)CCN(C(N2CCC(OCc3ccccc3)C2)=O)C1 C=CCCCCC(=O)N(C)CC1CCCN1C(=O)C(O)Cc1cccc(Cl)c1 c1(C(=O)NCCN(C(C2C(C)CCC2)=O)CCOCCO)cccc2occc12 c1(C(=O)NCC(C2CC2)NC(C2(CC=C)CC=CC2)=O)ccc2c(c1)ncn2C c1(CC)ccc(C(N2CC3CN(C(c4ccccc4C(C)C)=O)C3C2)=O)cc1Br c1(CNC(CCC=C)=O)cccc2c1CCN(C(=O)C(C)(C)c1nccs1)C2 N1(C(C(C(C)NC(CCOC)=O)(C)C)=O)CC2(C1)OC(=O)NC2C c1(CCC)nc(C)c(C(=O)NC2CCN(C(C3CCCN(C(C)C)C3)=O)C2C)o1 N1(C(C=Cc2n(C)ccc2)=O)CCC(C)(NC(=O)CC2CC(F)(F)C2)CC1 c1(C(C)(C)C)cc2n(n1)CCN(C(=O)Cc1cc(Cl)ccc1[N+](=O)[O-])C2 CC1(C)CN(C(c2ccc3[nH]ccc3c2)=O)CCC1NC(=O)COC1CCCC1 c1(CCC(=O)NCC(CCNC(C(C)Sc2ncccn2)=O)O)ccc(Cl)nc1 C1(C(=O)NCCNC(C2CC(=C)C2)=O)CSCN1C(=O)C(C)CC Cc1ncc(Br)c(C(N2CCOCC2CNC(C2(CO)CC2(F)F)=O)=O)n1 C1(CC(=O)NCC2(O)CCN(C(=O)C3CC3)C2)CCN(C(c2nccs2)=O)CC1 C(=O)(C1=C(C)CCOC1)NCC(C)(CO)CN(C(CNC(CCOC)=O)=O)C CCCC(C(=O)N1CCCC(N(CCO)C(c2c[nH]ccc2=N)=O)C1)OC O=C(CC(C(F)(F)F)NC(C1(CF)CC1)=O)Nc1cnc2ccnn2c1 C12(NC(CSC)=O)CCCC1N(C(C1(CCOCc3ccccc3)CC1)=O)CC2 C(=O)(C#CC(C)(C)C)N(CCCn1cc(COCCCCO)nn1)C CC1CN(C(=O)C(C)(C)c2cnsc2)CCC1NC(c1cc(N)c(F)cn1)=O C1(NC(c2csc(C3CC3)n2)=O)CCC2CCN(C(C3(Cl)CC3)=O)C1C2 C1(NC(CNC(CN(C)C2CC2)=O)=O)CCC1(C)C.C1C(=O)N1CC1CC1 c1(C(N(C)CC2CCN(C(C3C(C)C3)=O)C2)=O)cccc2c1OC(F)(F)O2 S(=O)(=O)(c1cc(C)cnc1NCC1COc2ccccc21)NC(C(CC)CC)C N1(C(c2c(C)ocn2)=O)CC2CC(NC(=O)C(C(C)C)c3cccnc3)CC2C1 c1(CC(N2CC(CC(C(=O)NC3(CC#C)CC3)F)C2)=O)ccc(C#C)cc1 C1(CNC(=O)Cn2nccn2)CCCC(CNC(C2(C(F)F)CCCCC2)=O)C1 Cc1noc(C)c1CC(N1CC(NC(c2ccnc(OC(C)C)c2)=O)C(C)C1)=O CC12COC(C(=O)NC3CCN(C(c4cccn4C4CC4)=O)C3C3CC3)(C1)C2 C(=O)(C(C)C(F)(F)C(F)F)N1CCC(C)(NC(CC2(CC)CCOCC2)=O)C1 N1(C(c2cncc(N)c2)=O)CCOC2(CCCN(C(=O)C(O)CC(F)(F)F)C2)C1 C1(C)(COC)CCCN1C(=O)CONC(c1ccc(C)cn1)=O c1(C(N2CCC3(NC(C4=CC(C)(C)C4)=O)C(C2)C3)=O)ccc(S(N)(=O)=O)c(F)c1 C(N=C(NCC1CC2C=CC1C2)NC1CCC1)C1CC(NC(N)=O)C1 c1(CC(C)NC(C2C(C(=O)OCC)C2)=O)ccccc1SC C1(NC(c2cc(C)nnc2)=O)CC2CCC1CN2C(=O)C(c1ccccc1)C c1(OC)ncnc(C)c1C(=O)NC(C1CCN(C(c2cnnn2C)=O)C1)C N1(CC(=O)OC(CC)C)CCN(CC(F)F)C(C2CC2)C1 C(=O)(CCCC(=O)NCC(C)CC(=O)NC1CNC(=O)C1(C)C)N(C)C Cn1cc(C(N2CC(NC(c3cc[n+]([O-])cc3)=O)C(F)C2)=O)nc1O C1(NC(CCCOC)=O)CCCC(N(C)C(c2nc(Cl)cs2)=O)C1 c1(OCC)ccccc1C(=O)NC1CC(C(N)=O)C1.C12CCN(C1)C(=O)CO2 C(CC(C(C)C)NC(c1nc(C2CC2)oc1C)=O)N(C(CNC(CCC)=O)=O)C N1(C(CCCOCC)=O)CCC(NC(=O)COCP(C)(C)=O)C(CC)C1 C1(C(N2CC(C)(NC(C3CC(OC)C(OC)C3)=O)C2)=O)CCC(C)(C)CC1 N1(C(C(C(C)(C)O)NC(C2CC=CCO2)=O)=O)CCN2CCCCC1C2 C1(CNC(Cn2c(C)c[nH]2)=O)CC2(CO1)CN(C(c1cc(C#N)on1)=O)C2 C(=O)(C(C)CNC(C1(CC)COC1)=O)NC(C#C)CC N1(C(=O)NC2CC2)CCC(OCC2(c3cccc(C(F)(F)F)c3)CC2)CC1 N1(C(C2CCN(C)CC2)=O)CC(C)(C(N2CCOC(C)C2CO)=O)CC1(C)C n1(CC(=O)N(C2CN(C(c3ccc(CC)[nH]3)=O)C2)C)ncccc1=O C1(C(=O)NCC(CC)NC(C2(c3ccccc3F)CCC2)=O)CC2C(C1)C2(F)F c1(C(N(C)CC2CCN(C(Cn3ccc(C)n3)=O)C2)=O)cc(C2CC2)nn1C c1(CNC(C(n2cc(CC(=O)OC)nn2)C)=O)c(CC(=O)OC)noc1C N1(C(Cc2cn(C)nc2)=O)CCCCCC1C(=O)Nc1cncc(Cl)c1 c1(CC(=O)NC(C)CNC(=O)COC2CCC2)ccccc1NS(=O)(=O)C1CC1 C1(CC)(CO)CCN(C(C2CCCC(CNC(C3CCC(O)CC3)=O)C2)=O)CC1 c1(CC)cc(C(N2CCC(NC(C34CCCC3C4)=O)C2C2CC2)=O)ncn1 C12(NC(COC3(C#C)COC3)=O)CC(CN(C(C3CCOC3C3CC3)=O)C1)C2 C(=O)(C1=NN(C2CC2)C(=O)CC1)NC1(CNC(C(c2cccc(C)c2)O)=O)CC1 CC(C)CC(O)C(=O)NCC12CC1CN(C(=O)C=Cc1cn(C)nn1)C2 N1(C(C(C)NC(C)=O)=O)CCN(C(=O)CC2(C)CC2(F)F)C(CC(F)F)C1 c1(CC)cc(C(=O)NCCCOCCNC(=O)CCCN(C)C(=O)OC)on1 N1(C(c2c(OC)ccs2)=O)CCC2CC2(C(=O)NC2CCCCC2C#N)CC1 C1(CNC(C(CC)COC)=O)CCN(C(=O)CCc2cnoc2)CC1CC CC(C)(C#N)CCC(=O)NCCNC(c1ccc(C(F)(F)F)cc1)=O Cc1ccncc1C1CC1C(=O)NCC1CN(C(=O)CCC2CC2)CCO1 Cc1cc(C(=O)NC(C2CN(C(C3CCC(=O)C3)=O)C2)C)n(C2CC2)n1 CC(CCC(C)(C)C)C(=O)NC1(C)CC(C(=O)N(C)CC2CC2)C1 C1(NC(C=CC(CC)=CC)=O)CC2CCC1N2C(=O)Cc1cnc(C)s1 C(=O)(C1=C(c2ccccc2)CCC1)N1CC(C2(NC(CCCC#N)=O)CC2)C1 c1(C(C)C)c(N2CCCC(CCNC(C3CCCC3O)=O)CC2)ncnc1Cl c1(N(C)CC2(OC)CCCOC2)ncc(I)c(C)n1 C(=O)(C1CCCc2sccc21)NC1C(NC(c2c(SC)cc(F)cc2)=O)COC1 c1(C(C(=O)NC(C2CN(c3nnc(CC)o3)C2)C)OC)c(F)cccc1F c1(CNC(C(CC)(C)F)=O)nnc2n1CCN(C(C1C3C4CCC(C4)C13)=O)C2 N1(C(CN2CC(CC)C2)=O)CCC2(CCC2)C(CNC(C2(O)CC(C)(C)C2)=O)C1 N1(C(CCCC=C)C(=O)NC(C)C)CCc2c(C#N)cccc2C1 c1(CC(=O)NC(CN(C(c2c(OC)n[nH]c2)=O)C)C)ccc(F)c(Br)c1 C(CC(O)CC(=O)NCC#CCNC(C1CCC(=O)NC1)=O)SC C1(NC(CCNS(CC)(=O)=O)=O)CCN(C(=O)CCC2CC(C)C2)C1 C1(C(=O)NC(c2cn(CC)nn2)C)(CF)CCN(C(=O)CC2CCCSC2)C1 C(=O)(C(C(C)C1CC1)N(C)Cc1ccco1)NCCCOC c1(C(=O)NC(CC)CN(C)C(C23CSCC2C3)=O)cnc(Cl)c(N)c1 c1(C(C)C)cc(C(=O)NC2(CNC(C3CCC(C)S3)=O)CCC2)no1 c1(C(N2CCN(C(c3cnc(C(=O)OC)s3)=O)CC2)=O)ccc2nc[nH]c2c1 C1(C2CC2)(C(=O)NC2CCC(CCNC(C3(C)CCC3)=O)C2)CCC1 C1(NC(Cc2c(C)noc2Cl)=O)CN(C(=O)COCCOC)C2(CCCOC2)C1 N1(C(C)=O)CCCN(C(C2CN(C(=O)C(C)(C)CC3CC3)CCN2C)=O)CC1 C1(C(=O)NCC2OCCN(CC)C2)N(C(=O)C=CCOC)CC12CCCC2 C1(CC(=O)NC(C2CCCCC2)C)CCCN1C(C1(n2cccc2)CCCC1)=O c1(C(N2CC(NC(C3(C=C)CCC3)=O)C(C)CC2)=O)cc(O)c2c(cnn2C)c1 C1(CNC(CC(COC)(C)C)=O)CCC(C)(C)CN1C(=O)CC12CCC(CC1)C2 Cc1nc2cc(Cl)cc(C(N3CCCOC(CNC(=O)CSC4CC4)C3)=O)c2[nH]1 C1(CNC(CNCC(=O)OC(C)(C)C)=O)CCN(c2ccc(Cl)cc2)C1=O N1(C(C2(OC)CCSC2)=O)CC2CC2(NC(=O)Cc2csc(C(F)(F)F)n2)C1 C(=O)(C1=CCC(F)(F)CC1)N1CC(C)C(CNC(c2ccc(=O)n(C)c2)=O)CC1 C#CCC(CC(=O)N(CCCCO)C)NC(=O)C(C)Cn1ccnc1 c1(C(=O)NC(c2ccc(OC(F)(F)F)cc2)C(=O)OC)c(I)ncn1C C1(F)(CNC(CCC(=O)NC)=O)CCCN(C(C2COCCN2CC(F)F)=O)C1 C1(CC(=O)N(C2CC=CC2)CC)C(NC(=O)Cc2cccs2)CC1O N1(C(CCCC(C)(C)C)=O)CCC2(CC1)CC(NC(c1ncsc1C1CC1)=O)C2 C12(CNC(C(C)OCCCC)=O)CN(C(=O)CC3(O)CCOCC3)CC1CCO2 C1(CC=C)(C(=O)N(C2CCN(C3CC3)C2)C2CC2)CCCN1C(=O)CCC(=O)N(C)C n1(CC)ncc2cc(C(=O)NC3CC3NC(=O)C(C)C(C)C)c(C)nc12 N1(C(c2c(C)cc(OC)nc2)=O)CC2=C(C1)CN(C(c1cscc1SC)=O)C2 Cc1cc(COC(C2CCCN2c2nnn(C)n2)=O)on1 c1(C(N2C(c3cn(CCOCC)nn3)CCC2)=O)coc2c1CSC2 N1(C(=O)OC(C)C)CCC(CN2CCN(C(c3ccc(Cl)cc3)C)CC2)CC1 C1(CC)CCCC1(C)C(=O)NCC(C(C)C)NC(C1CCCN1C1CCCC1)=O CCCC(F)C(=O)NCCC1(OC)CN(C(C2(CC3CC3)CCC2)=O)C1 C1(O)(C(C)NC(c2cc(-c3ccsc3)[nH]n2)=O)CCN(C(=O)CNC(N)=O)CC1 c1(NC(C2(CNC(c3cc(Cl)cnc3Cl)=O)CC2)=O)cccc2c1OCO2 C1(C(=O)NC2C(C)(O)CCC2)CC2C=CC1N(C(c1cn(C3CC3)nn1)=O)C2 c1(C(=O)NC(CC(=O)NCC(C)(C)N(C)C)C(F)F)c[nH]c2ccccc12 C1(C(=O)NCCCn2c(C)nnc2)CC(C)(C)CN1C(C1CC(=O)NC(=O)C1)=O c1(-c2n(CC=C)c(N3CCN(C(=O)COC)CC3)nn2)c(F)cc(F)c(F)c1F c1(C(=O)NCC2CC(C(=O)NC3CN(C)C3)C2)c(O)cccc1F C1(O)(CN(C)C(c2cnc(O)o2)=O)CCCN(C(=O)Cn2cnc(Br)c2)C1 C1(CC)C(C(=O)NC2CC(O)C2O)CCN1C(c1c[nH]nc1Cl)=O N1(C(c2c(C(C)C)ncnc2)=O)CCN(C(=O)C(c2cccnc2)C)C(C)C1 C1(CNC(c2c(C)cc[nH]c2=N)=O)CC2CCC1N(C(=O)C(F)(F)C1CC1)C2 Cc1ccc(C(=O)NC2CC(C(F)F)(NC(=O)Cc3ccc(O)nc3)C2)nn1 C1(C(=O)NCC(C)N(C(=O)CC2(n3ccnc3)CC2)C)CCCC2CCCN12 Cc1cncc(C)c1C(=O)NC1CCCN(C(C2(N(C)C)CCCC2)=O)CC1 N1(C(C2CSCC(=O)N2)=O)CCOCC(F)(CNC(C2(C(F)F)CCC2)=O)C1 C1(C(=O)NCC(C)N(C(=O)CSC(C)(C)C)CC)C2CCC(=O)C12 C1(C(=O)NCC2C(C(=O)OC)C2)CCN(C(c2cnc(Cl)s2)=O)C1 c1(C(=O)NCCN(C(CC(C)C)C)C(C2CC(O)C(F)C2)=O)ccc(CF)cc1 c1(C(N2CCC(c3ccnn3C)CC2)C(=O)NCC=C)cc(C)c(OC)c(C)c1 C(CCCCCCN)N(C(C(CC)Cl)=O)C c1(C(N2CCC3(C(NC(=O)CC4CC(F)C4)C3)CC2)=O)c[nH]c2ncnc(O)c12 C1(C(C)(C)C)CC2(CCN2C(C2CC3(CCCO3)C2)C(=O)NC2CC(F)(F)C2)C1 C(=O)(C(C(=O)NN(C(=O)CC(C)CF)C)OC)OCC.C1(C)(CO)CC1 N1(C(CCC#C)=O)CC2CN(C(=O)Cc3nncn3C(C)C)CC2(C)C1 C1(NC(C2(C=C)CCC2)=O)CC(C(=O)NC2COC(C(C)C)C2)CC1O c1(OC)c(O)cc(C(=O)NCC(C2CC2)NC(=O)CC(C)(C)C2CC2)cc1C#N Cc1cc(C(=O)NCC(C(C)C)NC(c2ccco2)=O)cnc1C(F)(F)F C1(NC(C2CC(C)CN(C(C3SCCS3)=O)C2)=O)C(=O)OC2CCCC12 CC(CS(C)(=O)=O)C(=O)N1CC2CC1CCC2NC(=O)CCCN1CCCCC1 c1(C(N2C3C(C(=O)Nc4ncc(F)s4)CC(CC3)C2)=O)n[nH]c2c1CS(=O)(=O)C2 CC1OCCCC1C(=O)NCC1C(C(=O)NCCN2CC(CF)C2)C1(C)C C1(NC(c2ccc(OC)nn2)=O)CCC(C)N(C(=O)Cc2cscn2)C1 C1(NC(=NC)NCCC2CC2(F)F)CC12CCOc1ccccc12 CC1Oc2ccc(C(=O)NCC3(F)CN(C(c4cc(=O)cc[nH]4)=O)C3)cc2C1C CC1(C)CN(C(C23CCCC2CN(C(=O)CC2CCOCC2)C3)=O)CC(C)(C)O1 c1(NC(C)=O)cc(Br)ccc1C(=O)NCC(C)(CO)NC(=O)C=CC1CCC1 Cc1nc(C)c(C(=O)NCCCOc2cccnc2)o1.C1CO1 C(=O)(C(C)(C)CCCOC)Nc1ccc(C(=O)NC(CSCC)C)cn1 c1(C2(C(=O)NC3C(NC(C(CCOC)C)=O)C3)CC2)ccc(OC)c(OC)c1 Cc1oc(C(C)C)cc1C(=O)NC1CC(C)(NC(=O)CNC(=O)C(F)(F)F)C1 C(=O)(CC(C(C)(C)C)NC(=O)CN1CCCCC1)NCC=C CC1(C(=O)NCc2ccsc2C(=O)NCc2nn[nH]n2)CC=CCC1 c1(N2CCC(C(C)NC(CCNC(COC)=O)=O)C2)ncnc2[nH]c(C)c(C)c12 Cc1cc(NC2CCOCC2F)ncc1S(=O)(=O)N1CCC=C(Br)C1 n1(CC(=O)NCC(C)NC(=O)CC2CCCCO2)c(S)nc2ccccc2c1=O Cn1ccc2sc(C(=O)NCC3CCCN3C(=O)CC3CCNC(=O)C3)cc12 n1(C(C)C(N2CC(F)CC2CNC(c2nocc2Cl)=O)=O)cc2c(n1)CCCC2 Cc1cccc(C(=O)NCCN(C(c2cccnc2C(F)F)=O)C2CC2)c1 c1(C(N2C(C(=O)NOCCCN(C)C)(CC)CCC2)=O)ccc(C#N)n1C c1(C(C)(C)C)cncc(C(=O)NCCCNC(=O)CCC2CCC(=O)N2)c1 N1(C(C2(SC)CC2)=O)C2CCC1C(F)C(NC(c1cc3c(=O)[nH]ccn3c1)=O)C2 N(C1CCCc2c[nH]nc21)C(C12CCN(C(C3CN(C(C)C)C3)=O)C1CCC2)=O c1(C(C(=O)NC(CCNC(CSCC)=O)C)C)ccncc1 c1(C(=O)N(C(CCC(=O)N2CC(c3onc(C)n3)C2)C)C2CC2)cnc2n1CCC2 OC1CC(NCC2CC2c2cccs2)C(O)C1 c1(C(=O)NCC2CCN(C(C(C(=C)C)(C)O)=O)C2)nc2n(c1Cl)CCCC2 C1(C(N2C(CC(=O)NCCCC(F)F)C=CC2)=O)C2CCC(F)(F)C12 c1(OC)ccc2[nH]cc(CNCC3(NC(=O)Cc4ccc(O)cn4)COC3)c2c1 c1(CC(C)NC(=O)CSCCNC(=O)Cn2nccn2)ncn(C)n1 c1(OCC=C)ccc(CN(CCC(C)(C)C)CCOC)cc1 C12(NC(CC(C)n3cccc3)=O)CC1CN(C(c1cc(Cl)ns1)=O)C2 c1(C(=O)NCC2(O)CN(C(c3c(C(C)C)noc3)=O)C2)c[nH]c2cccc(F)c12 C(C(C)(C)C(=O)N1CC(N(C)C)C(F)C1)N(C(=O)CCOCC(F)F)C Cc1ccc(C(=O)NC(CNC(C2CC2C)=O)C(C)C)c2c1NCCC2 C(=O)(C(C(=O)NC1(CC(=O)NCc2nccn2CC)CC1)OC)OCC N1(C(C(C)c2cncs2)=O)CC(F)(CNC(C2CC2c2ccccc2)=O)C1 Cc1coc2ccc(C(N3CCC(NC(C4CC5(F)CC4C5)=O)C(O)C3)=O)cc12 C(CNC(C1CC12CC2)=O)(CC(=O)N=c1cc(C)n(C)[nH]1)OC c1(C(=O)NCC2(O)CCN(C(=O)CC3C=CCC3)C2)cccc2ccsc12 N(C(=NCC1CC(OC)C1)N(C)Cc1ccsc1)CCSCC=C Cc1nc(C(N2CC(CF)(NC(=O)CC3OCCOC3(C)C)C2)=O)cn(C)c1=O C1(NC(N2CCCCC2c2ccccc2)=O)CCC([N+](=O)[O-])CC1 C1(C(=O)OCC(C2CCC(F)(F)CC2)=O)COc2cc(Cl)ccc2O1 N1(C(C=CCN(CC#C)C)=O)CC2(C1)SCCC2NC(=O)CSCc1cscn1 O=C(C1Cc2ccc(Cl)cc21)NC1CC2CCC1CN2C(=O)CSC1CC1 C(=O)(CCCC(=O)NCCC1CCCCN1C(C1CN(C(N)=O)C1)=O)NCCC C1(NC(=O)C=Cc2ccccn2)CCN(C(C2(F)CCCCC2)=O)CC1CO Cc1cc(C(=O)NCC(C)NC(=O)CC2(CO)CC2)ccc1-n1ccnc1 c1(C(=O)NCC(CC=C)NC(c2cnoc2C(C)C)=O)cncc2nc[nH]c12 Cc1cc(CNC(=O)N(CC(C)CCO)C)c(C)cc1Cl Cc1ccccc1C(C)CC(=O)NCC(C)NC(=O)C=CCN(C)C C1(NC(c2ccc(OC)nc2)=O)CC12CCN(C(=O)CCc1ccnn1C)CC2 N1(C(CC2N(C(CC(CC)SC)=O)CC(O)C2)=O)CC(S(C)(=N)=O)C1 C12(CC(=O)NCc3c(C)nn(C)c3)CCC1CN(C(c1c(C)csc1C)=O)C2 C(=O)(C1=C(Cl)CCC1)NCc1c(C(=O)NC2CCN(CC)C2)nco1 C(=O)(CC(C)CN(C)C)NC(C1CCN(C(C2CC(=C3CCC3)C2)=O)C1)C C1(CNC(C(CN(C(CC(CC)SC)=O)C)(C)C)=O)CC2(CCC2)CO1 c1(CN(C(=O)CC2CC3CCC23)C)ccn(CC(F)F)n1 c1(CC)ccc(OCC(N2CCC(CNC(=O)C(N)=O)C(C)C2)=O)c(Br)c1 C#Cc1ccc(Cl)c(C(=O)NCC2CCN2C(c2cc(Br)n(C)c2)=O)c1 c1(C(C)=O)cnn(C)c1N.C12(CC13CCC3)CNC(=O)C1CC(OC1)C(=O)NC2 c1(C(C)C)ccccc1C(=O)NCC1CN(C(=O)CSc2nnnn2C)C2CC12 N1(C(c2cccnc2SC(F)F)=O)CCCC(O)(CNC(C2(CO)COC2)=O)C1 c1(CC)occc1C(=O)NC(C)CCNC(C1(CN(C)C)CC1)=O C1(N(c2nc(N3CC4CCC3C4)nc3cc[nH]c23)C)COC2(CCOCC2)C1 c1(C(N2C3(CNC(=O)C4=C(Cl)CC4)CC(C2)C3)=O)cc2ccccc2nc1O CC(C(=O)NCC=CCNC(=O)COc1ccc(CC(N)=O)cc1)C(C)O N1(c2ccnc(NC(c3ccc(Br)cn3)C)n2)CCCC2(C=CCO2)C1 Cn1cc(NC(=O)CCN(C(c2cccc(CC#N)c2)=O)C2CC2)c(O)n1 Cn1ccc2cc(C(N3CCN(Cc4coc(C5CC5)n4)C(C#N)C3)=O)ccc12 N1(C(C2CC(C)C2)=O)CCCCC1CCNC(c1ncncc1N)=O N1(C(CC(C)(C)OC)=O)CCC2CCN(C(c3cc(C)nc(O)c3)=O)CC12 C1(C(N2CC3C(N(C(C(C)c4ccsc4)=O)C)C3C2)=O)CCC([N+](=O)[O-])CC1 c1(C(=O)NCC(COC)(C)O)cccc2ccc(O)nc12 CCCCCN(CCC(=O)NCC1(O)CC1)CC CN1CCCC(O)(CC(=O)NCC(C(C)(C)C)NC(=O)CC2CC3CC3C2)C1 CC1(NC(=O)Cn2ccnn2)CCN(C(C2(N3CCOCC3=O)CC2)=O)C1 O=[N+]([O-])c1cnn(CCNC(c2nnnn2C2CCC2)c2cnco2)c1 C(=O)(CC(C)C(C)(C)CC)NCCN(CCC)C(c1cnn(C)c1Cl)=O c1(OC(C)C)n[nH]cc1C(=O)NC(C)(C)CCNC(=O)CNC(c1cscn1)=O C1(CC)CN(S(C)(=O)=O)CCC1NC(=O)C=Cc1ccc(SC(C)(C)C)cc1 c1(C(c2nnnn2CCCF)NCCCSC)ccc(F)cc1SC C1(C(=O)NCCC2CN(C(C=CC(C)(C)C)=O)C2)CCC(NC(N)=O)CC1 c1(CN(C)CC2CCN(C(C)=O)C2)csc(=NCc2cccc(I)c2)[nH]1 C1(c2nnnn2C2CC2)(NCC2ON=C(C)C2)CCc2cc(Br)ccc2C1 c1(C(=O)NCC2N(C(CC3CC(=O)OC3)=O)CC(F)C2)cccc2sncc12 C(=O)(C1=NOC(CNC(C2CCC2C#N)=O)C1)N(C(C)C(C)(C)O)C N1(C(C2(C(=O)OC)CC2C)=O)CCC2(CC(NC(=O)C3=C(Cl)CCCC3)C2)C1 C1(C(=O)NC(CC(C)C)CNC(c2cc[n+]([O-])cc2)=O)CC(F)(F)CCC1(C)C c1(CCC(=O)NC23CC2CN(C(=O)CCn2ccccc2=O)C3)cccc(Cl)c1 C1(Cl)(C(=O)OC)CC12CCN(S(=O)(=O)c1ccc(C(C)(C)C#N)cc1)CC2 Cn1nccc1C(=O)NC1CC(C(N2CCCC2c2ccncc2)=O)C1 c1(C(=O)NCC(CNC(C(C)=CC)=O)OC)cc(F)cc(F)c1N NC1CC2(CC(C(=O)NCC(c3cnn(CC(N4CCCC4)=O)c3)=O)C2)C1 C(=O)(CCC(C)O)NC1CC(CNC(c2c(CCC)[nH]cc2)=O)C1 N12CCN(C(=O)C1)CC2=O.c1(OC)ncc(CNC(c2ccsc2)C)cn1 c1(C(=O)NC2C(C)CN(C(c3cc4ccsc4s3)=O)C2)ccc2c(n1)COCC2 CC1CC(C(=O)NCCCCCCNC(c2ccccc2-n2cncn2)=O)=NO1 Cc1cn(C2CCOCC2)nc1C(=O)NC1CC(F)(CNC(c2cnsn2)=O)C1 N1(C(C(C(C)C)c2cccnc2)=O)CCCC(NC(=O)C(C)n2cnnn2)C1C S(=O)(=O)(c1ccc(OCC(=O)Nc2cc(O)ccc2Br)cc1)NCC1CCCO1 c1(C(=O)NCC2(CO)CCN(C(CS(=O)(=O)NC)=O)C2)ccc2c(c1)CCC2 c1(C(N2CC(OC)CC2C(=O)OC)C(=O)NC)cc(Cl)cc(Br)c1F CCS(=O)(=O)c1cccc(C(=O)N(C2CCCN(C(c3ccnn3C)=O)C2)C)c1 c1(C(=O)NC2CCCN(C(C(C)NC(=O)C(C)(C)C)=O)C2)nnc(Cl)cc1N C1=CC2CC1CC2CN=c1nc(N2CCOCC2)[nH]o1 c1(C(=O)NC(CNC(CC(=C)Br)=O)(C)C2CC2)csc2cncn12 C1(C(N2CCN(C(Cc3c(C)non3)=O)CC(O)C2)=O)CCCC2CCCCC12 N1(C(c2n(CC(C)C)ncc2)=O)CC(NC(=O)CCc2ccco2)CCC1C CN1CCCCCC1C(=O)NCCCCNC(c1ccc(O)c(Cl)n1)=O c1(C2(C(N)CN3CCN(Cc4ccccc4)CC3)CC2)ccc(Cl)cc1 c1(C(N2CC(F)CC(NC(C(C)O)=O)C2)=O)cc(N)cc([N+](=O)[O-])c1 N1(C(c2c(C)nc(CC)o2)=O)CCC2CCC12CNC(c1cc(C2CC2)on1)=O N1(C(C(CC)(C)C)=O)CCCC(CCNC(=O)C(c2cccc(OC)c2)O)CC1 CC1CCN(C(=O)CC(C)(C)CNC(=O)C(F)F)CCS1 C1(NC(c2cc(F)cc(Cl)c2)=O)CC2CN(C(c3cc(O)cc(Br)c3)=O)CC2C1 CCC(CC(=O)NC1CN(C(c2cc(C3CC3)on2)=O)CC1N=[N+]=[N-])C(C)(C)C CCC(CCOC)C(=O)NCCOCCn1cc(CSC2CCOC2C)nn1 c1(CC(N2C(CNC(C(C(C)(C)C)=O)=O)CC(F)C2)=O)cnc2cccnn12 N1(C(C23CCC(OC)C2C3)=O)CCC(C=CC(N2CCCCCC2CO)=O)CC1 C(=O)(CC(C)(C)CNC(c1ncccc1N)=O)N(C(CC(CC)C)C)C Cc1cc(F)ccc1C(=O)NCCNC(C1CCCN(C2CCN(C)CC2)C1)=O C(=O)(CC(C)(F)F)NCCN(CC(C)O)C(c1cnn(C2CC2)c1Cl)=O C1(C(N(C(C)C)CCNC(c2cccn2C(C)C)=O)=O)CC2C=CC1C2 C1(CNC(C(C)C2CCC2)=O)C(C(=O)N(CC(O)CN(C)C)C)C1(C)C N1(C(c2cc(C)no2)=O)CCOC(CNC(=O)Cc2nncn2C(C)C)C1 c1(C(=O)NC(C2CCCCC2)CNC(c2cscc2Cl)=O)cncc(F)c1 CC1CN(C(C23CC(CCO2)C3)=O)C(C)CN1C(=O)Cn1ncc2ccccc12 C(=O)(C(C)(C)CCCNC(C1CCCC1C)=O)NC1(C(=O)NC(C)C)CC1 C1(C(=O)NC(CC)CN(C)C(C2(CO)CC2)=O)CCCN1CCCF CCC(C#N)(CC)C(=O)NC1CCCCC1NC(=O)C(C(C)C)NS(N)(=O)=O C1(C)(C(N(C2CN(C(c3cc(N)cc(O)c3)=O)CC2O)C)=O)CCN(C)C1=O c1(OCC(=O)NCCC2CCN(C(=O)CCc3cncnc3)C2)cccc(F)c1 C1(CC(=O)N(CCc2cn(C3COC3)nn2)CC)CN(C)CC1O C(=O)(CC(O)CC(C)(C)C)C(CC)CC.C1(CN(CC(=O)NC)CC)CCNC1 c1(CC(=O)NC2CCC2CNC(=O)CSc2nncs2)cc(O)nc(O)n1 Cc1ccc(CC(=O)NC2CC3C(NC(C4CCCSC4C)=O)C3C2)cn1 C12(C(=O)OC)CCNCC1CN(S(=O)(=O)CCOCC(F)(F)F)C2 c1(CNC(C2N(C(C3N(CC)CC3)=O)CC2)=O)cc(C2CC2)on1 N1(C(C(N2CCOCC2)C)=O)CC(C(=O)NCc2nc(C(N)=O)co2)C2(CC2)C1 c1(C(C(=O)NCCNC(c2cc(Cl)n[nH]2)=O)OC)cc(F)cc(F)c1 c1(C(=O)NC2CCC(CC(N3CCC(COCC)CC3)=O)C2)c(C)[nH]c(C)c1C c1(C(=O)NCC(CCOC)NC(=O)C2=CCCC2(C)C)cccc2cccnc12 C1(C2CCCO2)(C(=O)NCC2=CCN(C(CCN(C(C)=O)C)=O)CC2)CCCO1 CC(C)(C)CCC(=O)NC1C=CCN(C(C2CCCC3CC23)=O)C1 c1(CC)c[nH]nc1C(=O)NC1CC1CNC(=O)C(=O)N(C)C c1(NC(c2c(C)noc2C)C)cc(Br)ccc1[N+](=O)[O-] C1(C(CN(C(C)CC(=O)OC(C)(C)C)C(C)=O)F)CCCCCC1 C(=O)(CC(O)CC(C)(C)C)NC(c1ccc(C)cc1)CNC(CCC=C(C)C)=O C1(NC(C(C)ONC(=O)OC(C)(C)C)=O)CC2CC(C1)N(C(=O)CN(C)C)C2 N1(C(C(CC=C)(F)F)=O)CCCC(F)(CNC(=O)CC2CCCCC2(F)F)CC1 C1(CNC(C(CC)n2cccn2)=O)CN(C(=O)Cc2ncc[nH]2)CC1C c1(OC)cc(C(=O)NC2CCN(C(c3ccsc3C(F)F)=O)C2)cc(OC)n1 CC1(C(=O)NCc2cc(F)ccc2F)CCCN(C(C2CN3CCC2CC3)=O)C1 CCCCC(CCC)OC(c1conc1CC)=O CC(C)CC(F)(F)C(=O)NCC1CN(C(=O)CN2CCC(C)(O)C2)CCC1(C)C C1(c2cn(CCC(=O)N(CCCC)C)nn2)CCC(=O)CC1 C=CCCC(C(=O)N1CCCC(CO)C1)NC(C1CC1CC)=O C12(C(N3CCC4(O)CC4C3)=O)CCC(C(N3C(C(=O)O)CSCC3)=O)(CC1)CC2 C(=O)(C(CO)C(C)(C)C)N(CC(CNC(C1(C(C)O)CC1)=O)(C)C)C c1(OC)cc(C)cc(C(N2CCN(C(=O)Cn3cnnc3O)CC(O)C2)=O)c1C O=S(=O)(c1ccc(NC(CO)CCF)cc1Br)NCC1CCOCO1 C1(NC(COCC)=O)CCCCCC1NC(=O)C(C1CC1)SC c1(CNCC2N(C(c3cccc(C(N)=O)c3)=O)CCOC2)cc(Cl)ccc1Br Cc1[nH]nc2c(C(N3CC(NC(c4cc(Cl)c(Cl)cc4O)=O)C3)=O)cccc12 C1(NC(c2cc(C=C)cc(F)c2)=O)CC2CCC(C1F)N2C(c1csnn1)=O C1(C)(C(N2CC(C)N(C(c3ncccn3)=O)CC2)=O)CCCCC1(F)F c1(C(N2CC(C)(NC(CCC(C)SC)=O)C2)=O)cc(Br)cc(Cl)c1O c1(OC)c(C(N2CCCC(NC(C3CCCOC3C)=O)CC2)=O)cc(F)cc1F c1(C(=O)NC2CCC(CCNC(CCOCCCOC)=O)C2)cccc[n+]1[O-] c1(CCC(=O)NCCN(C2CCCCCC2)C(c2cc[nH]n2)=O)cncc(F)c1 CC1(C)CN(C(C23CC2CNC3=O)=O)CCC1NC(=O)CSC(F)F C1(N(C)C)CC2(CCC(C(N3CCC3CNC(=O)C3=CC4CCC3C4)=O)CC2)C1 N1(C(C(C)NC(=O)NC)=O)CCCCC(N(C(=O)C(=Cc2ccccn2)C)C)C1 c1(C(=O)NCC(C)CN(C(=O)CC2(C)CCC2)C)nn(C)c2ccc(F)cc12 C1(NC(c2ccsc2C(F)F)=O)COC2(C1)CN(C(C1CCOC1)=O)C2 Cc1cccc2c(CC(=O)NCCC3=CCN(C(=O)C(C)(C)CF)CC3)c[nH]c12 CCCC(C(=O)NC)NC(C1CN(C(=O)CC(C)n2cccn2)CCO1)=O C(=O)(C#CC1CCOCC1)NC(CC(CC)C)C(=O)NCC1(CC(N)=O)CC1 c1(C(=O)NC(C)CCNC(=O)CN2CCCNC2=O)ccc(Br)c(F)c1 N1(C(c2c(C)n(C)cc2)=O)CCOCCC1C(=O)NC(C)Cc1ccco1 c1(C(N2CC(C)C(NC(c3nc(Cl)sc3Cl)=O)C2)=O)cccn2cnnc12 c1(C(=O)NC2(CCNC(=O)CC3CC(F)(F)C3)CCC2)csc([N+](=O)[O-])c1 c1(CC)cccc(C(=O)NCC(CNC(=O)CCNC(=O)COC)CO)c1F N1(C(C(CC)(CC)CO)=O)CC(CNC(=O)CCc2nc[nH]n2)OC2(CCC2)C1 N=c1[nH]c(C2CC2)ncc1C(=O)NC1CC1NC(=O)Cn1nnnc1C1CC1 C(=O)(C(C)(C)C(C)(F)F)NCC1(OC)CCN(C(c2ncc(F)cc2F)=O)C1 c1(C)[nH]cnc1C#N.CCC(C)(CNC(=O)CCOCCOCCO)NC(C)(C)C C(=O)(C(C)(CNC(=O)CN1CCCC1)CC)NC1CON(CC)C1=O c1(OC)ncc(C(=O)NCCC(C)N(C(=O)CO)C)cn1 C1(C(=O)OC)CCOC(C)C1.c1(NC(N2CC(=O)NCC2)=O)ccc(Cl)cc1 N1(C(c2cc(F)c(CO)c(F)c2)=O)CCC2(CCN(C(C3CSCCS3)=O)C2)C1 N1(C(c2cc(CC)ncn2)=O)CCN(C)C(C(=O)NC2CCCOC2)C1 C1(NC(Cc2cccc(C)c2F)=O)CN(C(c2ccnnc2S)=O)C2(CCC2)C1 C1(NC(C(=O)NC2CC2)=O)CC2COCC2N1C(C1(c2ccccc2)CC1)=O C=C(C)C(C)(C)C(=O)N1CC(C(O)C(=O)N(C2CCN(OC)CC2)C)C1 c1(C(N(C)CC2N(C(CNC(C(CC)C)=O)=O)CC(F)C2)=O)nc(C)n(C)c1C C1(NC(c2cc[nH]n2)=O)CN(C(c2cc3n(n2)CCC3)=O)C2CCCC12 C1(NC(c2nc(Cl)sc2Cl)=O)CN(C(c2nccs2)=O)CC1(F)F C1(C(=O)OC)C=CC(C(=O)NCCC2(C)CN(C(c3c[nH]nc3OC)=O)C2)C1 c1(NC(CCC)=O)ccnc(C(=O)NCc2cc(C(=O)NCC)on2)c1 C1(C(N)=O)CC2(CCN2C(c2sccc2CNC(=O)CC2CCCC(=O)C2)=O)C1 C1(CCl)NC(=O)N(CCl)C2=C1C(=O)NC2C.c1(N(C)C)cc(Cl)cc2c1C(=O)O2 C(C(C)(C)CC(F)F)NC(C(n1cc(-c2cccc(CNC(C)=O)c2)nn1)C)=O C1(C(=O)NCC2(C)CC(NC(c3c(C)con3)=O)C2)CCCCN1S(N)(=O)=O N1(C(c2ncn(CC)n2)=O)CC2CC(C(=O)NCC3(CCOC)CC3)C(C2)C1 C1(C(=O)NCCCN(C)C(c2ncc(F)cc2N)=O)CC2(C1)CC1(CC1)C2 N(C1CCc2c(Cl)ccc(Br)c21)C(CC(C)(C)N(C1(C)CCOC1)C(c1ccco1)=O)=O C1(NC(CC2(OC)CCC2)=O)CC(NC(c2cn(C)nc2C)=O)C12CCC2 N1(C(C2C(NC(CC=C)=O)CCO2)=O)CCOCC1C(C)C c1(C(=O)NC2CN(C(C3C(CC)CCC3)=O)C2)cc2cccc(C)n2n1 N1(C(c2c(CCC)nco2)=O)CCOC(CC(=O)NC(COC)CCO)C1 CN1CCC2(CCN2C(=O)CC2CCCN(C(C3(O)CCSCC3)=O)C2)C1 N1(C(CC2CC(OC)C2(C)C)=O)CCC(NC(c2ccn(C)n2)=O)CC(C)(C)C1 CC1CN(C(C2COC(CNC(C34CC(C)(CCO3)C4)=O)C2)=O)CC1(C)CO c12ccc(C)c(c1)C(=O)NC1CC1CNC(=O)C2.c1(SC)cccc(C(N)=O)n1 c1(CC(N2CCCC(CNC(c3cc(C)c(C)s3)=O)C2)=O)ccc2c(c1)OCO2 N1(C(=O)C=CC(F)(F)F)CCCC2C(NC(c3cccc(OC)n3)=O)C(C)(C)C12 N1(C(COCCCC)=O)CCN(C(=O)C(C)CCO)CCC1C C1(S(N)(=O)=O)(C(=O)NC(C)C(CO)NC(=O)COCCF)CC1 C1(NC(c2cc(C)[nH]n2)=O)CC2CCC1CN2C(=O)CC1C=CCCC1 C(=O)(C1Cc2ccccc21)NCC(CNC(=O)C1=COCC1)C(F)(F)F CC1CCCCCC1NC(=O)CCCCNC(=O)CC1CCN(C)C1=O c1(N(C(C)CNC(c2ccc(C(C)(C)C#N)cc2)=O)C)ncnc2c1nnn2C c1(C(=O)NC(CNC(c2c(C)csc2)=O)C(C)C)cccn2nnnc12 n1(CC(=O)Nc2c(C(=O)NC(CC=C)CO)cc(OC)nc2)nnc2ccccc12 C1(NC(C(CC)CO)=O)CCN(C(=O)CSC2CC2)C12CCC2 CCC(C)CC(C)C(=O)NCC1(C(N2CC(O)(C(=O)OC)C2)=O)CC2(CC2)C1 C1(CN(C(C(C2CC2)OCC)=O)C)CCCCN1C(c1sc(SC)cc1C)=O c1(OC)ncc(C(=O)NC2CCCC2CC(=O)NCCC(C)C)cn1 c1(C(=O)OCC)oc(=NC(C)C2CCN(C(C)=O)CC2)[nH]c1C(F)(F)F C(CC(C)C(=O)NCc1ccc(CN2CCCC(C)C2)cc1)=CCC C1(NC(C(C)CS(C)(=O)=O)=O)CN(C(C2(C(C)(F)F)CC2)=O)CC2(CCC2)C1 Cc1cn2c(C(N3CCN(C(c4cnnc(O)c4)=O)C(C(F)F)C3)=O)cnc2s1 c1(C(C)=O)cc(C(N2CCN(C(=O)C(F)=CCCF)C(C(C)C)C2)=O)ccc1F c1(C(=O)NC2CC(NC(c3c(C)cc(Br)c(F)c3)=O)C2)ccnc2ccccc12 C1(NC(c2ccc(C)nc2)=O)CN(C(c2occc2C)=O)CC2(CC2)C1 C(=O)(CCC(CF)CF)N1CC2C(CC(=O)NC(C)(CO)C3CC3)C2C1 C1(CNC(C(C)(C)OC)=O)CC2COCC2N1C(C1(N(C)C)CCCCC1)=O C(=O)(C1=C(C)CCCC1)N1CCC(C(C)Nc2ncc(C(=O)OC)cc2Cl)C1 c1(C(N2CC(C)C(NC(=O)CN(CC(C)(C)C)C)C2)=O)cc(C#N)ccc1N C=C=CCCC(=O)N1CCC(O)(CCNC(C23CCC(CC2)C3)=O)C1 C(=O)(CCCCCCCC)NCCCCCC(=O)NCC(=C)F c1(CC(=O)NC2C(CNC(C3OCC(=O)NC3)=O)C2)c(Cl)cccc1Cl C1(C(=O)NC2C(NC(C=Cc3n(C)cnc3)=O)CCC2)CCc2cnn(C)c2C1 c1(OCC(=O)NC)ccc(CC(=O)NC2CCN(C(=O)C(C)N(C)C)C2C)cc1 CCCCCC(O)CC(=O)NC1CC(CCC(=O)NCC(C)CCO)C1 Cc1nccc(C(=O)NC(Cc2ccoc2)C(=O)NCC2(CO)CCC2)c1N CC(C)C(C)(CNC(=O)Cc1cccnc1C(F)(F)F)NC(=O)CC(F)F CC1CCC(c2nnnn2CCCF)(NC(c2nccs2)C2CC2)C1 CC1CC(C(N2CC(c3ccon3)C2)=O)CN(C(c2cnns2)=O)C1 CCCCC(F)(F)C(=O)NC1CC(C(F)C(=O)NCCCC2CCC2)C1 O=S(=O)(c1c(F)cc(Cl)cc1F)NCCCCc1cnc[nH]1 C1(NC(COC(C)=O)=O)CCCC1(C)CN(C)C(c1csc(-c2ccsc2)n1)=O c1(N(C)Cc2c(C)ccs2)ccc(S(=O)(=O)NCCc2nccnc2C)cn1 c1(C(=O)NC2CCC(C)(CNC(c3c(OC)csc3)=O)C2)cc(OC)cc(C)n1 C#CCC(CC(F)F)C(=O)N1CC(C(=O)Nc2cccc(C)c2)(COC)C1 N1(C(c2n(C)ccc(=O)c2)=O)CCCC(C2CN(C(=O)C3CC3)C2)C1 CN1CCN(C(=O)C=Cc2cccnc2)C(CNC(C2(CO)CCCO2)=O)C1 Cn1ccc(OCCNC(=O)NC2(c3ccccc3)CCCO2)n1 N1(C(c2n(CC)ncc2)=O)CC(NC(c2ccnc(F)c2OC)=O)CC12CCC2 CC(CC(=O)NC(CCF)C(=O)NCC1CC2CCC2C1)C(F)(F)F N1(C(C2(CCO)CC2)=O)CCCC(Nc2ncncc2Cl)CC1 C#CCCCCCC(=O)NC1(C2CCN(C(=O)C3=C(C)CCC3)C2)CC1 c1(C(N(C(CNC(C(C)Oc2ccccc2)=O)C)C)=O)cc(Cl)ncc1F c1(OC(C)C)ncc(C(=O)NCC2CCC(NC(c3ccns3)=O)CC2)cc1Cl C1(C(=O)NCCN2CCN(C(C(C)CCO)=O)CC2)CNC(=O)CC12CCOC2 Cn1cc(C(=O)NC(CC(N)=O)c2cn(-c3ccccc3)nn2)c(=O)c(Br)c1 c1(OC)[nH]c(=N)ccc1C(=O)NC1CC2CCC1(NC(=O)CC1CC(F)(F)C1)C2 c1(NC(C2C3CN(C(C4(C)CCC4)=O)C2C3)=O)cc(C#N)c(F)cc1Br c1(NC(C2CCN(C(c3ccncc3Br)=O)CC2O)=O)ccc(Cl)c(I)c1 c12nc3ccc(cc3s1)OC2.C1(OC)CC(OCC)C(O)C1.c12cnn(c1)OC2 N1(C(C2(CCNC(CCc3cn(C)nn3)=O)CCC2)=O)CCOCC(CO)C1 C1(C)(CNC(c2c(C(C)C)nns2)=O)CN(c2cc(Cl)ncn2)CCO1 c1(CSCC)cccc(C(=O)NC(C)CCNC(=O)C(C)(C)c2ccno2)c1 C1(C(=O)NCCn2ncc(CC)c2)CC(C)CCN1C(c1cc(C)c[nH]1)=O C1(CC(=O)N(CCCCNC(C2C(C)(COC)C2)=O)C)CCC2(CCCC2)CC1 c1(SCC)nccnc1C(=O)NC(C)CCN(C(=O)C(C)N1CCC1)C CN=c1nc(N2CCCC(NC(=O)NC)C2)[nH]c(=NC2CCOC(C)(C)C2)[nH]1 N1(C(C(CC=CCC)C)=O)CCCCC(C(=O)NCC2CC(CC)=NO2)C1 CCCC(C)(O)CNC(c1cnn(CCNC(=O)CNC=O)c1)=O C(=O)(C1CCc2ccc(Br)cc21)N(CCN(C)C(C1COC(=O)C1)=O)C N1(C(CCC)=O)CCC(C(=O)NC(C)C(=O)OCC2(CO)CCCCC2)CC1 C1(COC)CN(C(c2cc(C)ccc2O)=O)CCN1C(c1ncnc(C)c1C)=O Cc1nc2cc(C(=O)NCCC(C)NC(C3COC(=O)C3)=O)ccc2n(C)c1=O C1(CNC(c2ccc(CCC)cc2)=O)CC(F)(F)CN1C(c1cc(OC)ns1)=O C1(NC(c2n(C)ncc2C(F)F)=O)CCN(C(c2cnc[nH]2)=O)CC1F C1(NC(c2c(CC)onc2)=O)CCCCCC1C(N1CC(c2cnc(C)s2)C1)=O C=CCC(CC=C)C(=O)N1CC2(CCC2)CC1CNC(=O)Cc1cscn1 CC1(CNC(=O)C(O)C2CN(C(c3ccco3)=O)C2)CCC(O)CC1 CCC(Cc1ccccc1)CC(=O)N(CCCNC(=O)C(F)CC(C)C)C1CC1 C(c1cccc(Cl)c1Cl)=CC(=O)Nc1cccc(NC(C2CCC(F)C2)=O)c1 c1(C(=O)NCC2C(CNC(=O)C=Cc3ccccc3)C2)cccc2[nH]cc(Cl)c12 C1(C(N2CCC(CC(C)C)C2)=O)CCCN(C)C1.c12c[nH]nc1CONC2=O C(=O)(C(O)CC(F)F)NCc1c(CNC(CN(C(=O)OC)C)=O)cccc1 C=CCC(CNC(c1sccc1Cl)=O)NC(c1ccc(F)s1)=O c1(C(N2CCCC2C(C)C)C(=O)NCCCC(=O)OC)cnc(CCOC)nc1 C(C)(CN=c1[nH]c2c(c(=NCCCc3ncc[nH]3)[nH]1)CSC2)SC N1(C(Cc2n(C)ncc2)=O)CCC(C2CC2)C1C(=O)NCc1ccnn1C N1(C(CCOC(C)C)=O)CC(C(N2CC(C)(C)CCC2CO)=O)CCC1(C)C N1(C(C(CC)O)=O)CC(NC(=O)C=Cc2cc[nH]n2)C(O)C1 CC(C)CC(F)C(=O)NCCN1CCN(C(=O)C(C2(O)CCOCC2)(F)F)CC1 CC1(C)C=C(C(=O)N2CCC(C)(C(=O)NCc3c[nH]nc3C3CC3)C2)C1 c1(C(N2CCC(C)(NC(CCCC(=O)OC)=O)CC2)=O)cccc2c1CCO2 C1(N(C(=O)C=CC=C(Cl)Cl)C)CCCC(NC(=O)Cc2ccc(C(N)=O)nc2)C1 c1(C(N2CCCC(N(C(C(C(CC)O)C)=O)C)CC2)=O)cccn2nncc12 N1(C(c2c(OC)cccc2)=O)CC2CC(CNC(=O)CCOC3CC3)C1C2 c1(C(N(C(CCNC(C2(COC)CC2(F)F)=O)C)C)=O)ccncc1Cl C#CCC(C(=O)N(CCCC)CC)NC(C1CCN(CC)CC1)=O N1(CC(C(C)N)O)CC(Sc2ccc([N+](=O)[O-])cc2)Cc2ccccc21 CCC(C)CC(C(=O)Oc1cccc(C(C)(C)O)c1)NC(=O)OC(C)(C)C C1(NC(C2CCC(=O)N2)=O)CC2C(NC(=O)Cc3cccc(O)c3)C2C1 C1(NC(=O)Nc2c(C)nn(CCN(C)C)c2)CCc2ncn(C)c2C1 Cc1nn(CC(C)C)c(C)c1CCC(=O)N(c1ccc(Cl)cc1C1CC1)C1CC1 N1(C(c2c(C)n(C)nc2)=O)CCC2CC2(C(=O)NCc2ncoc2C(C)C)CC1 c1(C(=O)NC2C3CCN(C(c4cc(F)ccc4F)=O)C23)coc2c1C(O)CCC2 c1(C(=O)NCC23OCC(NC(C4C(CC)C4)=O)(C2)C3)cc(F)c(F)c(O)c1F C1(C(=O)NC2CCN(C(C3CCCN3C3CC3)=O)CC2)CC12CC(F)(F)C2 N1(C(c2ccc(C)c(C)n2)=O)CC2CCN(C(c3cc(F)cc(F)c3)=O)C2C1 c1(C(=O)OC)cc(F)cc(Cl)c1NC(C1CC2CC2N1C(=O)CC1(O)CCC1)=O c1(OC)cc(C)cc(C(=O)NCC2CCN(C(c3[nH]cnc3C)=O)C2(C)C)c1C O=C(C(F)C(F)(F)F)NCCCCC(CO)NC(=O)CCn1cc([N+](=O)[O-])cn1 Cc1nc(O)nc(S)c1C(=O)N(C(CNC(=O)CC1(O)CCCOC1)C1CC1)C c1(C(=O)NC2CC2CNC(C2(C3CC3)CC2)=O)ccc2c(c1)S(=O)(=O)NC=N2 C1(C(=O)OC(C)(C)C)(NC(c2c(C)nc(C(C)C)s2)=O)CC(O)C1(C)C c1(C(=O)NC2CC(NC(C(C(C)C)OC)=O)C2)cnc2n1CCC2 N1(C(C2(NC(c3ccc([N+](=O)[O-])o3)=O)C(C)C2)=O)CC2(C1)CC(C)(C)C2 C1(O)(CCNC(CN(C(C)C)C)=O)CCCN(C(c2cc(CO)[nH]n2)=O)C1 N1(C(C2C(OC)CC2)=O)CC2(CCN(C(=O)C=CCF)CC2)CC1C N1(C(C(C(C)C)C2CCC2)=O)CCC(NC(c2cc(O)ncn2)=O)C(F)C1 c1(CC(=O)NCCCCCNC(C(CC)F)=O)cccc(Cl)c1 c1(C(N2CC(COC)(CNC(c3nnc(C)s3)=O)C2)=O)c(C)oc(C)c1C C1(NC(=O)CC2CCSCC2)C=CCCC1CO.C12(CC1)C(=O)N2 c1(CN2CCC(CC(=O)NCC=C)CC2)c(C)nn(-c2nc(C)cc(O)n2)c1C N1(c2cc(OCC)ncn2)C2CCC1CC(NC(C1(C)CCCOC1)=O)C2 c1(C(C)=O)cc(C(=O)NC2CCCC(NC(=O)Cc3cccnc3)C2)cnc1C c1(C(=O)NC(CC)CN2CCN(C)CC2)ccn2cc(-c3ccccc3)nc2c1 C1(OC)C(C)C(N(C)C(=O)Nc2ccc(Nc3ccccc3)cc2)C12CCC2 C1(CCC)(NC(c2cc[nH]c(=N)n2)=O)CCN(C(=O)C(C(C)C)NC(C)=O)CC1 c1(C(=O)NCC2CC(F)(CNC(CC(CC)SC)=O)C2)cc2occc2s1 c1(OC)cc(OC)nc(C(=O)NCC#CCNC(=O)CC2COCC(C)(C)O2)n1 Cn1cc(C=CC(=O)NCC2CC2NC(=O)C(c2ccccc2F)(C)N(C)C)cn1 N1(C(c2ccc(C)nn2)C(=O)NC2COC2)CC2(C)CCC2(C)C1 N1(CC(=O)NCC(c2ccc(F)cc2)NC(CSC)=O)CCS(=O)CC1 C(=O)(C#CC(C)(C)C)N1CCN(CC2(NC(c3c(C)cc(CO)o3)=O)CC2)CC1 C1(NC(C(C(CC)C)C)=O)CCN(C)C12CCCN(C(=O)COC(F)F)C2 Cc1ccc(C(=O)N(C(C)CNC(=O)CCc2scnc2C)C)cc1[N+](=O)[O-] CCN(OC)C(=O)CNC(=O)CN(C(C1CCCCC(=O)N1)=O)CC1CC1 CCC(C)(C)C(=O)C(=O)N1CCC2(CC2)CC1C(=O)NC(C)C#N c1(C(=O)NCC2N(C(c3cn(CC=C)nn3)=O)CC(O)C2)cccc(NC)c1C C1(NC(c2c(C)cnc(F)c2)=O)CC2CCC(C1)N2C(C1CCOC1C)=O C1(C(=O)NCC2(CNC(=O)Cn3nc(C)cc3C)CC2)(OC)CCC12CCC2 CCC(C)CC(C)NC(C1CCC(CNC(c2nc(O)sc2C)=O)C1)=O c1(C(=O)NCCCO)cccc(-c2cccc(C(=O)N(CCO)C3CC3)c2)c1 O=C1NCCc2c(C(=O)NC3(CO)CCN(C(c4ccc(Cl)o4)=O)C3)cncc21 C1(F)(C(N2CC3C(NC(=O)COCC4CC4)(C3)C2)=O)CC12CCCCC2 N1(C(C2CC(OC)(OC)C2)=O)CC(C(=O)NCCc2cccc(F)c2)CC(C)C1 c1(NC(c2c(C)nns2)C)ccc(S(=O)(=O)NCC2(C)CC2(F)F)c(Cl)c1 C=CCC(CC(=O)NCP(C)(C)=O)NC(c1oncc1CC)=O CCC(C)CCCCC(=O)N1CC(O)(CNC(=O)C=Cc2ccccc2Cl)C1 c1(NC(C2(C)N(C(CC=C)=O)CC2)=O)ccc(C)nc1CO C1(C(N(C(C(=O)NCC2(CC)CCC(=O)N2)C)C)=O)CCC(C2CC2)C1 CC1CCN(C(c2c[nH]c(=S)cn2)=O)C1C(=O)N(C1CC2(CCC2)C1)C C1(NC(C=CC(C)C)=O)C2CC3C1C3C2C(N1CCCC(C)C1CCO)=O CC1(C)CC(C(=O)NCc2cncs2)CCN1C(C1CCCC1C1CC1)=O c1(NC(N2C(C)(CNC(CC(C)n3ccnc3)=O)CCC2)=O)cc(F)ccc1F C1(CNC(c2c(COC)ncs2)=O)C(C)CCCN1C(=O)Cc1cccnc1Cl Cc1c(C(N2CCCC2(C)CNC(c2cnc(O)o2)=O)=O)sc2cncn12 N1(C(C(c2c(C)cccc2C)C)=O)CCN(C(c2cn(C3CC3)cn2)=O)CC(O)C1 N1(C(CN(S(CC)(=O)=O)C)=O)CCCCCC1CNC(C1CC(=O)NC(C)C1)=O C(=O)(C(F)CC(C)(C)NC(c1c[nH]c2ccccc12)=O)N1C(C)CC1CO N1(C(=O)NCC2(OC)CCNC2=O)CCOCC2(C1)CC2(F)F C#CC1CN(C(C2CCOC2CNC(c2nsnc2O)=O)=O)C1 C1(NC(CN(C)C(N)=O)=O)CC(C(=O)NCC2C=CCCC2)CC1O c1(CC(=O)NCC2N(C(C=C(C)C)=O)CCC2C)c(F)ccc(F)c1Br c1(OC)c(C(=O)NC2CC2NC(=O)Cc2cnccc2Cl)cnc2ccccc12 C1(NC(c2cnc(C)o2)=O)CCCC1(C)NC(c1coc(CC2CC2)n1)=O CCCC(C(=O)N1CC(O)(CNC(C2CC2c2sccc2C)=O)C1)NC(C)=O C1(C(=O)Nc2ccc(OCCOC)cc2)CC12CCN(C(C1(Br)CCC1)=O)CC2 c1(C(N2CCN(C(CSCC=C)=O)C(CC#N)C2)=O)ccc2cccc(Cl)c2n1 CCC(CC(=O)N1CC(CNC(=O)CC23CCCC2C3)C1)CC(C)C c1(OC)cnc[nH]c1=NCCC(C)NC(c1c(C2CCC2)cnn1C)=O c1(C(=O)NCCCN(C(c2c(CSC)cccn2)=O)C)cc([N+](=O)[O-])ccc1O c12cc(C)ccc1C(=O)N2.N1(C(=O)OC)CC(NC(C)=O)C1 CCC(CC(=O)NC1C2CCC(C2)C1C(=O)NCCCC(C)(C)CO)C(F)F c1(SC)ccc(C(=O)N(C2CN(C(=O)C(O)C3CCC3)CC2O)C)cc1 C=CCC(CC(C)C)C(=O)NC1CC12CCN(C(=O)CC1CSCCO1)C2 c1(CC(C)C(=O)NC2CCC(NC(c3cnco3)=O)CC2)ccc([N+](=O)[O-])cc1 c1(C(N2CCCN(C(C3(C)CCC(=O)C3)=O)CC2)=O)cc2n(c1)CCOC2 C1(C(C)NC(C2(CN(C)C)CC2)=O)CN(C(c2cc[n+]([O-])cc2)=O)CCO1 c1(C(N2CCCCC2CNCc2ccc3[nH]ccc3c2)=O)cc(I)c(F)cc1Cl CCC(C)(CNC(C1CCCN(C(=O)Cn2ccnc2)CC1)=O)C(N)=O Cc1ccc(=O)n(CC(=O)N(C2C3CN(C(C4CC(F)(CF)C4)=O)CC23)C)c1 C(CN=c1[nH]c(=NCC(C)N2CCCCC2=O)[nH]c2c1COC2)NC(=O)NCC N1(C(CC(COC)(C)C)=O)CCC2(C=C(C(=O)NCC3CCCC(OC)C3)C2)C1 Cn1ccc2cccc(CNc3ncn(C)c3C(F)(F)F)c12 C1(C(=O)NCC2N(C(c3cc(Cl)ncn3)=O)CC2)CCC(n2cccc2)CC1 Cc1c(C=CC(=O)NC2CN(C(c3cn(C)nn3)=O)CC2C(F)F)cnn1C Cc1oc(C(=O)NCC23CC(CN2C(C2CCC(C)CC2)=O)C3)cc1Br C(=O)(C1CCc2scnc21)NCC1N(C(c2c(CC)nc[nH]2)=O)CCC1 N1(C(CSCC)=O)CCN(N2CCCC2Cc2ccccc2)CC1 C(=O)(CC1CNc2ccccc21)NCC(C)(C1CC1)NC(C1CCSCC1)=O CC(C)C(C)(O)CNC(C1CCC1NC(=O)Cc1cn[nH]c1)=O C12(NC(CCS(C)=O)=O)CCCC1CN(C(=O)CC(C)(C)C#N)C2 N1(C(C=C)=O)CC2CC(N(C(=O)CCc3ncc[nH]3)C)C1C2 CCCC(C)CC(=O)N1CC2CC(NC(=O)C(C)(C)n3cc(Cl)cn3)C1C2 Cn1ccc(=NC(=O)C(F)Cl)cc1C(=O)OC(C)(C)C N1(C(C(CCC)OCC)=O)CCC(C=CC(=O)NCC23CCC(C2)OC3C)CC1 C=CC(CC)C(=O)N1CCSCC1C(=O)NOCC(C)O CCCC(CCC)CCN=c1ccn2ncc(S(=O)(=O)NCC3CC3)c2[nH]1 c1(C(=O)NCC(CNC(c2onc(C)c2C(F)(F)F)=O)O)nccc(Cl)c1C N1(C(C2(C#C)CC2)=O)CC(N(C)C)C(CNC(=O)CC2(OC)CC2)C1 c1(C(N2CC3CC3(CNCc3cc[nH]n3)C2)=O)ccc(Cl)nc1Cl N1(C(Cc2nc3scc(C)n3c2)=O)CCN(C(=O)OC(C)(C)C)CCC12CCC2 C1(NC(c2ccc(C(C)C)s2)=O)CC12CCN(C(c1ccoc1)=O)C2 n1(CC(=O)NC2CCN(C(c3c(C)cnn3C)=O)C23CC3)nnc2c1CCCC2 C1(C(N(CC(C)N(C)Cc2ccccc2)C)=O)CCCCN(C)C1=O n1(CC)ncc2c1CC(C(=O)OC(C)C(=O)Nc1ccc([N+](=O)[O-])cc1)CC2 N1(C(C(CCC)N(C(N)=O)C)=O)CCCC(C(=O)NCCOCC)(CO)C1 c1(N2CC(C)C(NC(=O)CC3(C(F)(F)F)CC3)CC2)ncc(Cl)cc1[N+](=O)[O-] C(C(C)(O)CCC)NC(COC1CN(C(CC=CCC)=O)C1)=O Nc1cc(F)ccc1C(=O)NCC1(F)CC(NC(c2scnc2C2CC2)=O)C1 c1(CCC(=O)NC2C(NC(CCC=CCC=C)=O)COC2)cc(C)sc1C C1(CC(=O)NCC(O)CNC(c2ccc[n+]([O-])c2)=O)CCC2(CC2)CO1 C1(NC(C23CC(NC(C(C)OCOC)=O)(C2)C3)=O)CCn2nccc2C1 C1(C(N(CC(=O)NC2CC2c2cccnc2)CC)=O)CCN(C(C)=O)C1 C1(CC(=O)NC)CCN(C(=O)C(N2CC(OC)CC2CSC)=O)CC1 Cc1cc(C(N2CCN(C(=O)C3=CCC3)C3CC23)=O)c2nc(C)n(C)c2n1 c1(-c2c(SCC(N3CCC(C)(NC(C(C)C)=O)C3)=O)noc2)ccc(F)cc1F Cn1ncc([N+](=O)[O-])c1CC1CCN(CCC2CCCC23CC3)C1 c1(C(=O)NCC2CCN(C(c3nc(C)oc3)=O)C2(C)C)c(C)nc(C(C)C)nc1O C#CCCCCCC(=O)N1CC(N(C)C(c2ccnc3[nH]cnc23)=O)C1 c1(OC)cccc(C(C)C(=O)NCC2CCC(NC(c3cnsc3)=O)C2)c1 C1(C(=O)OC)CC2(CCCC2)CN1C(c1ccc(OC(F)F)c(Cl)c1)=O N1(C(CCc2nc(C)sc2)=O)CCC2(CCC2)C(NC(=O)C2=CCOC2)C1 C1(C)(C(c2nnnn2CC2CC2)NCCC(=O)NC(C)(C)C)CC2(C1)OCCO2 CC(C)CCCC(C)C(=O)N(C1CCCN(C(c2ccc(N)cc2Cl)=O)CC1)C c1(C(=O)NCC2CN(C(c3cc(CC)c(CC)o3)=O)C2)cnn2c(C)ccnc12 c1(OC)ccc(NC(C2CCC(C)N(C(=O)CCC=CC(C)C)C2)=O)cc1C N1(C(C(CCCC)NC(=O)C=Cc2ccccc2)=O)Cc2ccncc2C1 CON(CCC(=O)N1CCc2ncn(C)c2C1)C(=O)CCC1CC(C)C1 C1(O)(C(CC)C(=O)NCC2(O)CC(CNC(=O)COCC(C)C)C2)CCCCC1 C12(CNC(C3CCCC(NC(C(C)NC=O)=O)C3)=O)CCC(CC1)OC2 c1(C(C(=O)NC)N(C)Cc2cnc(Cl)cc2C)ccc(Cl)c(Cl)c1C N1(C(C(C)C#N)=O)CCC(C)(C(=O)NCc2nn[nH]n2)C1 Cc1ccccc1COCC(=O)NC(C)CC(C)NC(=O)C(C)(C)C#N C(c1cccc(Cl)c1)=CC(=O)NC1(C)CCN(C(=O)COCC(F)(F)F)C1 N1(C(CCC=CC)=O)CCC(F)(CNC(=O)CC2CCN(OC)CC2)CC1 N1(C(CCn2ccc(C)n2)=O)CC(NC(c2ccn(C)n2)=O)CC12CCOC2 C1(C(=O)NCCC2(OC)CN(C(=O)CC(C)N3CCCC3=O)C2)CCCCC1O N1(C(C(C)OC)=O)CCC2CCCN(C(=O)CC3(O)CCCC3)C2C1 C1(COC(c2ccc(N3CCC(C)CC3)cc2)=O)CC(c2cccc(F)c2)=NO1 N1(CC(=O)N(CC=C)CC=C)CCC2(CCCCN(C(=O)C(CC)CC)C2)C1 c1(C(CNC(CCc2c(CC)cccc2)=O)C)cc(F)ccc1Br C1(CC)CCN(C(=O)NC(C)Cn2cc(C3CC3)nn2)C1NC(=O)OC(C)(C)C c1(CC)nc2sc(C)cn2c1C(N1CC(NC(=O)C(COC)COC)C(O)C1)=O N1(C(CNC(C)=O)=O)CCCC(F)(CNC(c2cccc(OC(F)F)n2)=O)C1 C1(NC(CNC(=O)OC)=O)CC2CCC1N(C(=O)Cc1ccnc(OC)c1)C2 C1(C(=O)NC(C)CN(C)C)CC(N=[N+]=[N-])CN1C(c1cnnn1C)=O C1(CNC(=O)CCCC2CCCC2)CN(C(=O)C=CC2CCCC2)CCO1 C(=O)(C1SCCc2sccc21)NCC1N(C(C=C(CC)C)=O)CCC1(C)C C(=O)(C1=CCC(F)(F)CC1)N1CC(CCCNC(Cc2cc(C)on2)=O)OCC1 c1(CC(=O)N(C)CC2CCN(C(c3c(C)cccn3)=O)C2)nc(F)c(F)cc1F c1(C(=O)NC2(CN(C(c3cc(C)oc3C)=O)C)CC2)ccc(F)c(Br)c1 C1(CC(=O)N(CCC)CCNC(=O)C(C)Cn2ccc(C)n2)CCCOCC1 c1(C(=O)NC2CC2)cc(Br)c(C)c(Br)c1.n12cc(C#N)cc1C2C.C12CC1NC2=O c1(C(=O)NC2CC(NC(C3C=CCC3)=O)C2)cnccc1C1OCCO1 c1(OC)ccc(Br)cc1NC(C1CCN(C(c2cccc(O)n2)=O)CC1)=O NS(=O)(=O)CCCC(=O)N1CC(O)(CNC(C2C3COCC23)=O)C1 CN=c1cc(C(=O)NC2CCCCC2CNC(=O)COCCF)cc[nH]1 c1(CC(=O)NCCCNC(C(CCO)N(C)C)=O)ccc2cc(O)ccc2c1 C1(NC(C2C(C)C2)=O)CCN(C(=O)C(O)CC2CCCCC2)C12CC2 C(=O)(CC1C(=O)Nc2ccccc21)NC1CCN(C(C2(OC)CC2)=O)C1 C1(NC(CNC(=O)NC)=O)CC2CN(c3cc(C4CC4)ncn3)CC12 c1(C(=O)NCC(C)CN(C)C(C2CCC2C(F)F)=O)csc(CC(F)(F)F)n1 Cc1cc(C(=O)NC2CC(NC(=O)CC3CCCOC3)C2)nnc1O c1(C(C(=O)NCCN(C(=O)C(C)c2ccsn2)CC)C)ccc(F)cc1F Cc1cc(C(=O)NCC2CCN2C(=O)CC2(CO)CC2)sc1-c1ccc(F)cc1 CC(CC(=O)N1CCCC1c1ccc(Br)s1)C(F)(F)C(F)(F)F c1(CC)nn(C2CC2)cc1C(=O)N(C(C)CCNC(=O)CCc1cn(C)nn1)C C(=O)(C(C(C)NC(c1ccc(C)c(C)n1)=O)C(C)C)NCCSCC c1(CNC(CC2(C(=C)F)CCC2)=O)ccc(CNC(=O)CC2CSC2)c(F)c1 c1(C(=O)NC2(C)CN(C(C3(C)CCC(C)C3)=O)C2)cnc2c(c1)COC2 c1(C(N(C(C)C)CCNC(=O)C(F)(F)C(C)O)=O)noc2ncccc12 N1(C(c2c(N)ccc(C)c2)=O)CCOCC(C)(CNC(C2CN(C(N)=O)C2)=O)C1 c1(CC)nc(CCC2(c3nnnn3CC(C)(C)CCOC)COC(C)C2)sc1C C1(NC(c2cnn(CCC)c2C)=O)CC2C1CCN2C(=O)C=CC1CCCC1 c1(C(N2CCC(NC(CC(C)c3ccco3)=O)C2)=O)cc(F)cc2nc(S)[nH]c12 C12(C(=O)NCCOCCN(C(C3C(C)C3C)=O)C)CC3CC(CC(C3)O1)C2 C(=O)(CC(O)CC(C)(C)C)N1C(C(=O)Nc2ccc(OC)nc2)C(C2CC2)CC1 c1(COC)ccccc1C(=O)NC(C)(C)C(C)NC(=O)CC(O)CN(C)C N1(C(c2c(F)ccc(C)n2)=O)CC(C2CN(C(C3(C(C)(F)F)CC3)=O)C2)C1 C12CCCN1C2.c1(CN(C)CCN(C(=O)Cc2nc[nH]n2)C)ccccc1 c1(OC)ccc(F)c(C(=O)NCC(C(C)(C)C)NC(C2C(C)OC(C)C2C)=O)c1 N1(C(C(=Cc2ccncc2)C)=O)CC(N(C)C(C2C=CCCC2)=O)C(C)(C)C1 CCCCCCC(=O)N1CCC(C(C)NC(C2(C)CCC(=O)NC2)=O)C1 c1(C(=O)NCC(C)N(c2cc(C(C)C)ncn2)C)cncc2ccsc12 N1(C(C2CC(C)(CC)C2)=O)CCCCC1CNC(C1C(C(C)=O)C1(C)C)=O c1(OCCOC)ccc(Br)cc1S(=O)(=O)N1CCC(c2ccccc2)C(C)C1 C(=O)(C(C(C)NC(=O)CC1(N(C)C)CC1)C(C)C)NCCC(=O)NCC#C C12(NC(C(C)CO)=O)CCCC1N(c1ccnc(-c3cccc(Cl)c3)n1)CC2 CN1CC(NC(=O)C(=O)NCC2C3CCC(C3)C2(C)C)CC12CCCC2 c1(C(CNC(C(C)SCC)=O)NC(=O)CC2CC(OC)C2)ccc(CC)cc1 c1(C(N2CCCN(c3scc(C(N)=O)n3)CC2)=O)cc(I)c(I)c(I)c1 c1(C(N2CCC(CC(=O)Nc3cccc(I)c3)C2)=O)c(O)cccc1F c1(OC)ccc(C(=O)NC2CC(CNC(c3cc(F)c[nH]3)=O)C2)cc1 n1(CC(=O)NCC2N(C(C3C(C)C3)=O)CC2)cc(NC(=O)OC(C)(C)C)nn1 c1(CCC)c(C(=O)NC(C)CN(C)C(c2cc(C)n(C(C)C)n2)=O)cnn1C c1(C(N2CCCC(CNC(C=NOC)=O)C2)=O)cccc(N=[N+]=[N-])c1 c1(N2CC(C)(N(C(C(c3ccccc3)OC)=O)C)C2)cc(Cl)nc(C2CC2)n1 c1(NC(C(=O)NC2C(CNC(c3cccc(C)c3)=O)CC2)=O)cc(F)cc(F)c1 C1(COC)(CNC(=O)CC2CCCC2)CCN(C(=O)C(C)N2CCCC2)C1 c1(C(N2C(C(=O)Nc3cnc(C)nc3)CC(O)C2)=O)cccn2nccc12 c1(CC(CC)C)nc(Cc2ccccn2)n(CCCN(C)C)n1 C1(C)(C(=O)OC)CN(C(c2ccccc2-n2cc(C(C)N(C)C)nn2)=O)CC1C Cc1ccc2c(C(=O)NC3(C)CCCN(C(C4CC(C)C4)=O)C3)onc2c1 CC1OCCN(C(C2CC(=O)CC(=O)C2)=O)C1C(=O)NC1CCCOC1 C1(C(=O)NCC2CN(C(C3(CCCC)CC3)=O)CC2(C)C)CCc2nncn2C1 N#Cc1cccc(C=CC(N2CCC(NC(=O)CCc3cncc(F)c3)C2)=O)c1 CC#CCCCC(=O)NC1CN(C(=O)CC(O)C(C)C)CC1(C)C c1(NC2CCN(C(CN(C3CC3)CC)=O)CC2C)ccc([N+](=O)[O-])cc1C(F)F c1(C(=O)NC(c2nc(C(=O)O)n[nH]2)CC)cc2n(n1)CCOC2 c1(NC(C2(CC)CC2(F)F)=O)cccc(CNC(C2CCCN2N=O)=O)c1 C1(C(N2CC(CC)N(C(c3ccn(C)c3C)=O)CC2)=O)CCCC(F)(F)CC1 CC1(C)CC(O)(C(N2CCC2CCC2C3CCCC23)=O)C1.c12cn(nn1)CC21CC1 C#CC1(C(=O)NCCCCCN(C(=O)CCc2cnccn2)C(C)C)CCC1 c1(NCc2ccnc(SC)n2)cc(F)c2cc[nH]c2c1.N12CCCOC(C1)C2=O N1(C(C)C)CCCC(C(=O)NC(C)(C(=O)NC(C(C)C)C2CC2)C2CCC2)C1 N1(C(c2c(C#N)ccs2)=O)CC2(CC(C(N3CC4(CNC(=O)N4)C3)=O)CO2)C1 CC1(C)CC(CN)N(C(=O)C2CC2)C1.c1c(Br)cccc1Br N1(C(C2(CC)CNC(=O)C2)=O)CCN(CCO)C(C)C1.N12CCC(C1)CCC2=O N1(C(C2CN(C)C(=O)C2)=O)CC(C)(C)C(NC(=O)CC(C)(F)F)C(C)(C)C1 CC1(C)OC(=O)CC1C(=O)NC1(C)CCN(C(C2(N=[N+]=[N-])CC2)=O)C1 c1(OC)cc(C)c(C)cc1-c1cc(NCc2cc(C)ccn2)ccn1 C1(CNC(c2c(C)cccn2)=O)N(C(=O)CCN2CCOCC2)CCCC1(C)C C1(CNC(C(CC#C)C)=O)CCC12CCN(C(c1nn(C)c(C)c1Cl)=O)CC2 C1(F)(CNC(c2c(-c3cn(C)nc3)cco2)=O)CCC(NC(c2cn[nH]c2)=O)C1 C1(C)(C(=O)NCC(C)NC(c2cc(OC(C)C)ncc2)=O)COC(C)(C)CO1 CC1(CNC(C2CC(=O)CN2C(C2CCSC2)=O)=O)CCCC1O CCCC(C)(CCC)C(=O)NCC(C)CN(C(=O)CCc1ccnc(Cl)c1)C N1(C(C(C2CCOC2)NC(CCP(C)(C)=O)=O)=O)CCCC(C2CC2)CC1 C1(C(=O)NCC(C)NC(c2ccc3nn[nH]c3c2)=O)CCC2(CCCCC2)CC1 CN1CCN(C(c2ccc(-c3ccccc3)o2)=O)CC1CNC(C1CCCO1)=O C=C1CCC(C(=O)NCC(=C2CN(C(C3CCC(O)C3)=O)C2)F)CC1 Cc1ccc(C(=O)NCC2(CCNC(C3COC4COCC34)=O)CC2)c(F)c1F c1(C(=O)NCCCC2(NC(c3cocn3)=O)CC2)nn2cccnc2c1Br C(=O)(C1=Cc2cc(F)ccc2OC1)N1C(C(C)NC(C2(C=C)CCC2)=O)CCC1 N1(C(c2cn(SCC)nn2)=O)CCOC2(C1)CN(C(c1c(C)cncc1F)=O)C2 c1(OC)cccc2cccc(C(=O)NC3(CO)CCN(C(=O)CC(C)F)CC3)c12 O=C(CS(=O)(=O)Cc1ccccn1)NCC1(NC(=O)Cc2cnns2)CCOC1 Cc1cc(F)ncc1NC(=O)CN(CC(C)C)C(=O)Cc1ccc(C#N)cc1 C(=O)(C(C)(C)N(c1ccncc1)C)NCC(=O)N(C(C)(C)CNC(=O)C1CC1)C N1(C(C2CN(CC)C(=O)C2)=O)CCC(O)C(N(C(=O)CSC(F)F)C)C1 C1(CNC(C2N(C(C)=O)CCCC2)=O)CCCN(C(c2sc(C)cc2Cl)=O)CC1 CON(C)C(=O)CNC(=O)CC(C)(C)N(C)C(c1ccnnc1O)=O N1(C(C(CC)OC)=O)CCC2CCCC12C(=O)NCCCCNC(=O)OC N1(C(c2cc(C)sc2-n2cccc2)=O)CC2CN(C(c3cscn3)=O)CCC12 c1(OC)cc2c(cc1Br)CCN(C(N1CCCC(O)C1C)=O)C2 Cc1cccc2c(C(=O)NC34CC3CN(C(=O)C(=O)NC3CC3)C4)csc12 C(C(=O)NC(CO)CCC)(C(C)CC)NC(COCCCC)=O c1(C(=O)NCC2(F)CN(C(C3(C)CC3F)=O)C2)ccc2c(c1)CCCC2 C(=O)(C1=CC2CCC(C1)C2)NC(C1CC(NC(C2(SC)CC(O)C2)=O)C1)C c1(C(=O)NC(CNC(C2(OC)CCCC2)=O)CC(C)C)cc2c(cc1O)CCC2 CC(CCCNC(C1CC(C)(C)C1)=O)NC(=O)C(C)(F)c1ccon1 CCCC(CC(=O)NC(C)CN(C(=O)CCC(C)(C)F)C)NC(=O)OC(C)(C)C C(=O)(CC1=CCN(C)CC1)N1CCCC(C(COC)C(=O)NCc2cccs2)C1 c1(C(=O)NC(COC)C)cccnc1C(=O)NCc1cnn(C)c1SC C1(CNC(c2n[nH]cc2F)=O)CCCCN(C(=O)Cc2cnns2)C1 C1(NC(c2ncc(OCC)nc2)=O)(CC)CCN(C(=O)Cc2cnsc2)CC1 C1(C(N2CCCC(C(=O)NC(C(C(=O)OC)C)C)C2)=O)CC(=O)N(OC)C1 c1(C(C(=O)N(CC(C)NC(=O)CC2C=NN(C)C2=O)C)(C)C)ccc(F)c(F)c1 C1(NC(=O)OC(C)(C)C)(CNC(N2CCOC(C3CCCOC3)C2)=O)CC(C#N)C1 N1(C(C(C(C)C)O)=O)CC2(CCC(CNC(=O)COC3CCCC3)O2)C1 C1(NC(C(COC)(C)C)=O)C2CC3C1C3C2C(N1CCOCC(O)C1)=O c1(CN(C(CCCCC)=O)C2CC3CC2CN3)ccc2nonc2c1 N1(C(C)C(=O)OCCCN=[N+]=[N-])CCC(c2ccnc(Cc3nn[nH]n3)c2)CC1 C1(NC(=O)CCC2CCCO2)CC2(C1)CC2NC(c1cc(C2CC2)on1)=O C(C)(C(=O)NC1COCC1CNC(c1ccn(C)n1)=O)(C1(C)CC1)OC c1(C(N2CCC(NC(C3(N(C)C)CCC3)=O)C2C2CC2)=O)ccc(F)c(Br)c1 c1(NC(C(C2CC=CCC2)N)=O)ccc2[nH]cc(Cl)c2c1 n1(CCN(C(C(C)C)=O)C)cc(CC2(C(=O)O)CN(Cc3ccccc3)C2)nn1 CCCC(O)(CCC)CC(=O)NCCCC(C)NC(=O)C(=Cc1ccco1)C N1(CCC(=O)NC(CCCC(=O)OC)C)CCc2ccc(OC)cc2CC1 N1(C(C(C)(CO)NC(CCc2n(C)ccc2)=O)=O)CCOCC(C)(C)C1 CC(CCCCNC(=O)CC1CCC1)NC(C1CCC(=O)N1CCC(F)(F)F)=O Cc1cnc(C(=O)NCC(CO)NC(c2cc(C(C)C)on2)=O)nc1 C1(C(=O)OC)CC2(CCC1NCC(=O)CC1CN(C(=O)OC(C)(C)C)C1)CC2 C(=O)(N=c1ccn(CCF)[nH]1)C1(C(C)C)N(C(C(C(CC)C)O)=O)CCC1 C1(CNC(C2(C(=O)OCC)CC2C)=O)(NC(C2CCCSC2)=O)CCOC1 C1(CC)CN(C(=O)C(CC)(CC)OC)CCC1NC(=O)Cc1c(C)cccc1F C(=O)(C(CC(F)F)NC(C1CCCC(=O)N1)=O)NCCc1c(C)ncs1 C1(CC(C)NCCn2cc(-c3ncoc3C3CC3)nn2)COc2ccccc2O1 c1(C(=O)NC(CN(C(c2ccccc2Br)=O)CC)C)cccc([N+](=O)[O-])c1 N1(C(C2CCC(C(=O)OC)C2)=O)CC2(CCN(C(c3cnc(C)s3)=O)CC2)C1 N1(C(CCOCCCOC)=O)CCN(C(C2CC23CCSCC3)=O)CC1C1CC1 N1(C(=O)C=CC2CCCO2)CCN(C2CCN(C(C3(Br)CC3)=O)C2)CC1 C(=O)(N1CCCc2nccn21)C1C(CNC(C(C(C)(C)O)F)=O)CCO1 c1(NCc2c(Br)cn(C)n2)[nH]c(=NCCCc2nc(=N)[nH][nH]2)nc2sccc12 C1(C(N(C(C)C)CCO)=O)CCCN1C(=O)C(C)C1CCCC1 c1(COC(C)C)nc(-c2ccn(C(C)C)n2)n(C2CCCc3ccccc32)n1 N1(C(c2c(C)nn(C(C)(C)C)c2)=O)CC(NC(c2csc(Cl)c2)=O)CC12CCC2 c1(C(N2CCC(NC(C(C)=C(C)C)=O)C(C)C2)=O)cccc2c1OCCN2C C1(CCC)(NC(=O)C(=O)NN2CCCC(C)C2)CCCN(C(=O)CC(F)F)C1 CC1CC(=O)NC1C(=O)NCC(C1CC1)NC(C1(C(F)F)CCCC1)=O N1(C(C(C=C)O)=O)CCC2(CCC2NC(=O)CCOCC(F)F)CC1 c1(OCC)ccc(C(=O)OC)cc1.C1(N(C)C)CCN(C(=O)Cc2cnn(C)c2)C1 C1(CNC(C(CSC)OC)=O)CN(C(=O)C(C(C)C)NC(C)=O)CCC1(C)C Cc1nc(=N)[nH]cc1C(=O)NC1CC(C)(CNC(=O)CCc2ccccc2Cl)C1 CC1CCC(CNC(c2nccc(C(C)C)n2)c2nnnn2C2CCCC2)CC1 C1(C(N(C2CCCN(C(C3CC(C)(F)C3)=O)C2)C)=O)CCC2(CC1)CC2(F)F c1(C(C(=O)NCCOC)N(C)CC2(C#N)CCC2)cc(Cl)c(F)c(Cl)c1 CN1N=C(C(=O)NC2CS(=O)(=O)CC2NC(=O)C2=CCCC2(C)C)CCC1=O C=CCC(C)(C)C(=O)NCC1CC(NC(=O)C=CCN2CCOCC2)C12CCC2 N1(C(C(C)OCC)=O)CCCC1C(C)NC(c1ccc(CN(C)C)[nH]1)=O C1(NC(=O)COCC2CCCCO2)CN(C(c2cc3scnc3[nH]2)=O)CCC1F C(CNC(=O)Cn1cnnn1)(C(C)(C)C)NC(c1c(CC)scc1)=O C1(CCNC(=O)COc2cccnc2)CC(F)(F)CN1C(C1C=CC=CC=C1)=O N1(CC)C(=O)CCC1C(=O)N(C(C)CN(C)C(c1cc(CF)on1)=O)C CC1(C)CCCC(CCNC(=O)Cc2ccsc2Cl)C1 N1(C(c2sc(CC)c(C)c2)=O)CCC(NC(C2CC3CC3C2)=O)C1(C)C c1(C(=O)NCc2c(C(N(CC(=C)C)CC)=O)[nH]cc2)cc(F)n(C)n1 c1(-c2ccn(C)c2)ccc(CNCc2cccnc2N2CCCCC2)cn1 c1cc2cc(-c3cn(C4CCCNC4)nn3)ccc2cn1 CCC(CC(=O)NCC1CCCC2(CC2)C1)N(C)C(c1cc([N+](=O)[O-])c[nH]1)=O O(N(CC)C(=O)CN(C(C1CC(=O)C1)=O)CC)CC c1(NCC(CCCC)NC(c2ocnc2CC)=O)ncc([N+](=O)[O-])cc1Cl N1(C(C(C)NC(c2ccoc2)=O)=O)CC(NC(=O)C(C)(C)CO)CC1CO C1(N2CCOCC2)(N(CC)CC)CCN(C(=O)C(N2CCN(CC)CC2)=O)CC1 C1(C(N2CCCC2C(C)C(=O)OC)C(=O)NCC(=C)C)COC(C)C1 O=C(C1CCc2ccccc21)NCC(O)CNC(C1CCn2cncc2C1)=O N1(C(CCc2cn(C)nn2)=O)CCC(C)(C)CC1C(=O)NCC(C)(C)C(C)(F)F C(=O)(CC(C)(CC)C(=O)OC)N1CCN(CCNC(C(CCC)=CCC)=O)CC1 C1(C(=O)NCCC2CN(C(C3CCCC3O)=O)C2)CC2C=CC1CC2 Cc1ncncc1C(N1CC(OCCC(N2CCC(C(C)O)C2)=O)C1)=O C12(CNC(CC(COC)C)=O)CC(NC(c3cc(C(C)C)nn3C)=O)(C1)C(C)O2 C1(CNC(C(Cc2c(C)nc[nH]2)O)=O)CCC(NC(c2cc(C#N)cs2)=O)CC1 c1(C(=O)NCC(CNC(c2nnc(C(C)(C)C)s2)=O)O)ccc(F)c2ccoc12 N1(C(C(C=C)(C)O)=O)CCC(O)(C(C)NC(=O)CCCOCC)CC1 C12(CNC(C3CC3F)=O)CN(C(c3ccnn3-c3ccccc3)=O)CC1CCO2 c1(C(N2CCC(NC(c3ccc(C(C)=O)cn3)=O)C2)=O)sccc1S(N)(=O)=O C1(CNC(CN(CC)CC)=O)CN(C(=O)Cc2cc(C(=O)OC)cs2)CCC1C C1(C(=O)NCC2CC(NC(CS(C)(=O)=O)=O)C2)CCC2(CC1)CC2(F)F c1(OCC(=O)N(CC(c2n(C)ncc2)O)CC(F)F)nc(O)nc(O)n1 S(=O)(=O)(c1cc(Br)cc2cccnc12)NC(C1CCc2ncc(Br)n2C1)=O Cc1cnc(C(=O)NCC2CC3CN(C(C4(n5ccnn5)CC4)=O)CC23)cc1C C(=O)(C1=CCCCC1C)N(C(C)CNC(=O)Cc1ccc(C)c(Cl)c1)CC N1(C(=O)NCC2(SC)CCOCC2)CCC2(CC(C#N)C2)C1 Cc1cc(C(N2C3CCC2CC3)C(=O)NC2CC2)c(C)cc1Br c1(C(N(C(C)C(=O)N(C)CC2(CO)CCC2)CCC)=O)sc(C)cc1C N12CCc3cc(ccc31)-c1cn(nn1)CC2=O.c1(OCC)ccc(F)c(Cl)c1Cl Cc1cc(Br)cc(C(=O)NC2CCN(C(=O)CCC(F)F)CC2CO)c1C Cn1ncc(Cl)c1C(=O)NCC1CC1CNC(c1cc(Cl)ns1)=O c1(CC(=O)NCC(=C)CCNC(c2cnc(OC)nc2)=O)c(C)nc(O)nc1C c1(CN(CCC)CCOC(=O)C(F)(F)C2(OC)CCCC2)ccccc1Cl C1(CC#C)(C(=O)NCCC(C)C=C)CCN(C(=O)CC(C)CC)C1 C(C(CNC(=O)CCSc1ccccc1)CO)NC(C)=O.c12cncn1NC2=O N1(C(C(C)(C(C)C)NC(C)=O)=O)CC2CCN(C(=O)C(N)=O)C2C1 N1(C(C2(NC(=O)Cn3cnnc3O)CC(O)C2)=O)CC(C2CC2(F)F)C1 C1(C(C#C)C)CCN(C(=O)CC(CC)N(C)C(c2cc(C)c(C)o2)=O)CC1 N1(C(CCNS(C)(=O)=O)=O)C2CCC1CN(C(c1cc(F)ccc1O)=O)C2 Cc1ccc(Br)c(CC(=O)NCCCNC(C2CC23CCSCC3)=O)c1 c1(OC)cccc(CC(O)C(=O)NC(C)CN(C(=O)CC(C)c2ccco2)C)c1 C1(C(=O)NC2CC(N(C(=O)CN3CSCC3=O)C)C2)CCOC2(CCCCC2)C1 C(C(=O)NCCCN(C(=O)CC1CCC(O)C1)C(C)C)(C(C)C)OC c1(CCNC(C(CNC(c2cc(C(N)=O)[nH]n2)=O)O)=O)cccc(F)n1 C(N=c1[nH]c(N(CCC(C)C)C)nc2ccsc12)C1(CCOC)CCC1 C(=O)(C1=CCC(C)CC1)N(CC(CNC(C1(OCC)CCCC1)=O)C)C C(=O)(C(C(=O)N1CCCC(N(C(=O)CNS(N)(=O)=O)C)C1)C(C)C)OCC C1(O)(CNC(c2cscn2)=O)CCCN(C(=O)CC2CC3CCC2CC3)CC1 c1(C(=O)NC(CC(C)NC(C=C(CC)CC)=O)C)cc2c(OC)cc(F)cc2[nH]1 C(CCCCCNC(C1C2CC2C2CC12)=O)N(C(=O)C=Cc1cccn1C)C c1(C(N2C(CNC(c3ncn(CC)n3)=O)CC2)=O)cc2cccc(OC)c2o1 Cc1cc2sc(C)c(OC(C)C(=O)OCC(C)C(C)CC(C)C)c2cc1[N+](=O)[O-] c1(C(=O)NCC(CNC(=O)C=Cc2ncc(C)[nH]2)OC)sc2nccnc2c1N C1(N(C=O)CC2CC3CCCCC3O2)(C2CC2)COC2(CCOCC2)C1 C1(CNC(=O)C(O)C2CCC2)CCCN(C(=O)CC23CCC(CC2)C3)C1 Cc1noc2ncc(C(=O)NC(CNC(c3ccc(S(C)(=O)=O)s3)=O)CO)cc12 CC1=C(C(=O)NC(C)(C)C(=O)NCCCOC(F)(F)F)SCCO1 C(C)(CC(C)(C)C)NC(C(C)N(C(=O)COCCCF)C)=O C(=O)(C(C)(C)C(N)=O)NCCCN(CCCNC(c1c(C)nc(C)o1)=O)C C(CC(C(C)(C)C)NC(c1ncc(C(F)F)s1)=O)N(C)C(C1CCC(=O)NC1)=O N1(C(CC(CC)C2CC2)=O)CCCN(C(C2(c3cccc(C#N)c3)CC2)=O)CC1 c1(C(=O)NCC2CC2NC(C2CCCCC2)=O)cncc2c(Cl)cccc12 Cc1ccc(Cl)cc1C(N1CC(NC(=O)C(O)Cc2ccccn2)C(C)C1)=O c1(C(N(C2CN(C(=O)C3=CC(C)(C)C3)CC2F)C)=O)ccc2nnnn2c1 c1(CC2N(C(C)=O)C(C)CCC2)cc(-c2cccc3c2OCC3)c2n[nH]cc2c1 c1(C(N2CC3(N(C(C4(C)CC4(F)F)=O)CC3)C2)=O)ccc2cnoc2c1 C1(C(N2C(CNC(CC3CC(C)C3)=O)CC(C)(C)C2)=O)COc2ccccc2O1 c1(OC)ccc(C)c(C(=O)NC(CNC(=O)CC2CC(C)=NO2)C2CC2)c1N c1(NC(CCCN2C(=O)CC(NC(C3CC(C)OC3)=O)C2)=O)cccc(Cl)c1Cl CC(CC(=O)NC1(C)CC(NC(=O)C(C)(C)C2CCCCC2)C1)C1CCCCC1 c1(OC)ccc(C(=O)NCC2(NC(C3COC(=O)C3)=O)CCCC2)cc1C(F)F C1(CNC(CC2(OC)CCC2)=O)(CO)CC12CCN(C(C1(C)CCCC1)=O)CC2 c1(OC)ncc(Cl)cc1N(c1ncc(I)cn1)C(C1CNCCC1(F)F)=O N(C1CN(c2ccc(C#N)cn2)CCc2ccccc21)C(CCC)=O Cc1[nH]c2ccc(C(=O)NCCN(C(=O)C(C)(C)CF)C3CC3)cc2c1C c1(C(N2CCC(C#N)C2)C(=O)N(C2CCCCC2)CC(F)F)ccc2c(c1)COC2 C(=O)(C(CC)C(C)C)NCC1(C(=O)NC(C(=O)NCC)CC)CCCC1 C1(N(C(C(=O)NCC)=O)C)CCC(NC(c2csc(COC)n2)=O)CC1 c1(C(N2CC(C)N(C(c3ccccc3F)=O)CC2)=O)cc(Br)cc2c1OCO2 Cc1c(C(=O)NCC2CN(C(=O)CCC3CCC3)CCCO2)cnc2ccnn12 CCC(C(=O)N(CCn1cc(C(N(C)C2CC2)C)nn1)CC)C1CCCCC1 CC1CCN(C(CC2(C)CCOC2)C(=O)NCCN2CCOCC2)CCS1 c1(C(N2CCC(N(C)Cc3cc(C)c(F)cc3)C2)=O)cccc2cc[nH]c12 CN1CCC(CC(=O)NCC2(NC(=O)CC3CCN(C)C3=O)CCOC2)CC1 N1(S(=O)(=O)CCc2ccccc2)CCC2(CCCC2N2CCCC(O)CC2)CC1 C1(NC(CC(=C=C)C)=O)CCN(C(=O)C(C(C)(C)C)N2CCCC2=O)CC1(C)C C1(CC(=O)NC(C)(CNC(c2cnn(CCO)c2)=O)CO)SC2=NCCN2C1=O Cc1cc2[nH]c(C(=O)NCC3(NC(=O)CCc4cnc(O)[nH]4)CC3)cc2s1 c1(C(=O)Nc2c(C)nsc2)ccc(F)c(S(=O)(=O)NC(c2ccccn2)=O)c1 Fc1cccc(C(C2CC2)NCC2CC2C2CCCC2)c1Cl c1(C(C(=O)NCC2C=CCN2C(c2ncccn2)=O)O)ccc(Cl)c(F)c1 C(=O)(CCCC(C)(F)F)NC(C(C(C)C)NC(c1ccc(C)c(C)c1)=O)C c1(Cn2cc(C(CCC)NC(c3cn(C)cn3)=O)nn2)n[nH]c2c(Cl)cccc12 N1(C(C(C)c2ccco2)=O)CC(O)CC1CNC(C1COC(=O)O1)=O C12(NC(CCCNC(N)=O)=O)CCCC1N(C(=O)CC1CNC(=O)O1)CC2 C12CCCCC1N(C(C1(C)C=CCC1)=O)CCNC2=O.CN(C)C(=O)N(C)C CCC(CC)CC(=O)N1C(CC(=O)NCC(C)CN(C)C)C2CCCC12 C1(OCCNC(C2(OC)CCSC2)=O)CCN(C(=O)C(C)c2ccsn2)CC1 c1(C(=O)NC(C2(C(=O)NCC3(CO)CCOC3)CC2)C)ncccc1O C1(CC(=O)NCCCC(C)NC(c2[nH]cc(C)c2)=O)CCCC2(CCC2)O1 C1(CC#C)CCN(C(C2(OC)CCN(C(c3ncn(C)c3C)=O)C2)=O)CC1 O=C(C1=CCCCO1)NCCCN(C(c1csnc1Br)=O)C1CC1 c1(C(N2C(COC)CN(C(C3(C)CC=CC3)=O)CC2)=O)cc(C)cc([N+](=O)[O-])c1 c1(C(N(CC(O)CNC(=O)CN(C(N)=O)C2CC2)C)=O)ccc(-c2ccco2)[nH]1 C(=O)(C(O)CC(C)(C)C)N1CCC(O)(CNC(COc2cccc(C)c2C)=O)C1 c1(C2CN(C(=O)OC(C)(C)C)C2)cc(NC(C(=O)N(C(C)CC2CC2)C)=O)n[nH]1 N1(C(COC)=O)CCC(C)C(N(C(=O)Cc2ccccc2NC(C)=O)C)C1 C1(C(=O)NCC2C(N(C)C)CCC2)CC12CC(NC(c1cnnn1C)=O)C2 CC(C(=O)NCC1CCCN1C(=O)CCn1ccnc1)C(C)O C1(C(=O)NCCC(CC)C)CCC(CNC(=O)CCCn2ccnn2)CC1 N1(C(c2c(C)ccc(C)c2)=O)CC(C(N2CCCOCC2)=O)C2(CCC2)C1 c1(CN2CCC(O)(C(=O)NC(c3ccc(C(C)C)cc3)C)C2)cc(F)cc(Br)c1 C(=O)(C(=O)N=S(C)(C)=O)N1CCC(=CCNC(c2nc(C(C)C)oc2)=O)CC1 S(=O)(=O)(c1cccnc1)NC1C(C(=O)Nc2ccc(OC)nc2OC)C1 C1(OC)COCCN(C(=O)CC2CN(C(C3CC4CCC(C3)C4)=O)C(C)(C)C2)C1 c1(NC(c2cn(CCNC(C3CCCC(=O)C3)=O)nc2)=O)ccc2ncccc2c1 CCC(CN(C)C)C(=O)N1CCC(N(C(=O)Cc2cnn(C)c2)CC)CC1 C1(CCNC(C2CC3CCC2O3)=O)CC2CCC(C1)N2C(c1cc(=O)cc[nH]1)=O C(=O)(C(C)(O)C(F)(F)F)N1C(C(N(OC)CCO)=O)CC2CC21 C1(CNC(CSC)=O)(NC(c2nc(Cl)sc2Cl)=O)CCC(C)(C)CC1 c12cccc(c1)C(=O)NC13CC(C1)(C3)NC2=O.c1(C2(C)CC2)cc(C(=O)O)on1 c1(C(c2nnnn2CCC2CC2)NC(CC)CS(C)(=O)=O)ccc(F)cc1Br CCC(C)(CO)C(=O)NCC1CCC(CNC(c2nn(C)c(C)c2Br)=O)CC1 C1(N(C(=O)CC2CCC2C)CC)CCC2(CC2)N1C(=O)CC1CCCCO1.CCC Cc1cccn2ncc(C(=O)NC(C3(CNC(=O)CC4(N(C)C)CC4)CC3)C)c12 C1(C(=O)NCC(COC)(F)F)CCC2CCC1N2C(=O)Cc1cc(C)no1 C(C(=O)OC(C)(C)C)(C(=O)N1CC(NC(=O)Cc2ccc(Cl)nc2)CC1C)OC c1(C(=O)NC(C(C)NC(c2c(C)nc(C3CC3)s2)=O)CO)c(N)cccc1F c1ccc(C(CC2CCCO2)NCCCc2cn[nH]c2)cc1 c1(CN(c2ncc(C)c(C)n2)C2(CN)COC2)c(F)cc(I)cc1F C(CC(C)C)(C(=O)NC1CN(C(=O)COC2CCCC(C)C2)CC1(C)C)OC Cc1cc(NC(c2cn(C)nn2)C)ncc1S(=O)(=O)NC(CO)CC(C)(C)C C1(NC(C2(COC)COC2)=O)CN(C(c2cccc(C)c2C)=O)CC2CC12 Cc1nc2cncc(C(=O)NCC3(C)CC(F)(F)CN3C(c3ccoc3)=O)c2[nH]1 c1(OCC(=O)NCCC(C)N(C)C(c2cccs2)=O)cccc(F)c1 c1(C(N2CCN(C(c3cc(C)no3)=O)C3(C2)CC3)=O)ccc2c(=N)[nH][nH]c2c1 Cc1cc(CNC(=O)C(C2CCCCC2)O)oc1C(N1CCC(O)(CO)C1)=O N1(C(C2C(C(=O)OCC)C2)=O)CCC(CCCCCNC(c2cnn[nH]2)=O)CC1 C(=O)(C(F)(F)C(F)F)NC(C(C(C)C)NC(c1snc(O)c1Cl)=O)C c1(NC(C2N(Cc3cc(C)c(Cl)nc3)CC2)=O)c(Cl)cc(Cl)cc1C#N N1(C(c2c(COC)cccn2)=O)CCCC(O)(CNC(=O)Cc2ccsc2)CC1 c1(C2CCN(CCC)CC2)nc(C2CCc3nnc(C)n32)n(C(C)C)n1 C(=O)(C1=CCCCC1C)N1CC(O)(CCNC(C(C(=O)OCC)C2CC2)=O)C1 c1(C(N2C(C)CN(C(C3CN(C4CCOC4)C3)=O)CC2)=O)cc(F)c(F)cc1F C1(NC(=O)CO)CC2CC(C1)N(C(c1cnn(Cc3ccc(Cl)cc3)c1)=O)C2 Cc1nc(-c2cccc(CN3CCCCCC3)c2)[nH]c(=N)c1F C(=O)(C(COC)CC(C)C)N1CCCC(CNC(Cc2c(CC)cccc2)=O)C1 C1(C(=O)NC2(CC=C)CCOC2)CC(=O)N(CNC(C2CC(F)(CO)C2)=O)C1 c1(CN(c2n(CCC=C)c(C(c3c(C)noc3Cl)C)nn2)C)c(F)cccc1Cl c1(CC)nc(C(=O)N(CC(C)N(C(=O)CCN2CCC2)C)C)cs1 c1(C(=O)NC(C)CCNC(c2ccc(F)c(C#N)c2)=O)ccnc2c1ccn2C c1(OC)cc(COC)ccc1NCc1ccc(OCCO)nc1 C1(NC(C2CC3(CC(C#C)C3)C2)=O)CCC2CCN(C(c3cccn3C)=O)C1C2 C12(C)CCCC1C2.N1(CC(=O)NN(C(CN(C2CC2)CC)=O)C)CSCC1=O CS(=O)(=O)c1ccc(C(=O)NCCC2CC(F)(F)CN2C(=O)C2CC2)s1 N1(C(C2CC(SC)C2)=O)CCC(C)(C)C1CNC(=O)C=CCN1CCCC1 C12(C(=O)NC3CCCN(c4nccc(C(F)(F)F)n4)C3)CCCCC1C2(F)F c1(CC)nc(C)c(C(=O)NC(C)(CNC(C2CCC(N(C)C)CC2)=O)CO)s1 C1(C(=O)NCc2ccc(SC)o2)CCN(C(c2ccc(F)c(O)c2)=O)C12CC2 CC1CN(C(=O)CN2C(=O)CCC2=O)CCC1N=c1cc(C(N)=O)nc(Cl)[nH]1 CC(C)CC(C(=O)NC1CCN(CCCO)C1)N(C(=O)CC1NC(=O)NC1=O)C N12C(CC3CC13)C(=O)Nc1scnc1C2=O.C1(COCC2CN(CC)C2)CCOC1 N12CC(C)CCC1OCCCC2=O.C(=O)(CSCC)NCCOCCOC C(CC(=O)N1CCN(CCNC(c2cc(C#N)n(C)n2)=O)CC1)(C(C)C)OCC C12(C(=O)NCC3(OC)CN(C(=O)C=C(C)C(F)F)C3)CCC(CC1=O)C2 Cc1cc(C(=O)NC(C2CCN(C(=O)Cn3c(C)ccc3C)C2)C)c(O)nc1C N1(C(C2CC(N(C)C)C2)=O)CCCC2(CCN(C(=O)COC3CC=CC3)C2)C1 C1(C#N)(C(N(CCC(C(C)C)N)C)=O)CCOCC1.C(CCC=O)=C(C)C N1(C(C(C=C)(C)O)=O)CCN(C(c2cnc(COC)s2)=O)C(CO)C1 C1(C(=O)OC(C)C(=O)Nc2ccc(F)cc2Cl)CCc2[nH]nc(O)c2C1 CC(C)(CNC(C1(c2cc[nH]n2)CC1)=O)CNC(C1(F)CCCC1)=O c1(C(N2CCC(NC(c3c(O)cc(C)nn3)=O)(CF)C2)=O)scc2c1OCCO2 CC(C)C(O)C(F)(F)C(=O)N1CCN(C(c2cn(C3COC3)nn2)=O)C(CF)C1 N1(C(C2(CCC)CC(=O)C2)=O)CC2(CC(NC(C3C4CC5C(C4)C35)=O)CO2)C1 c1(C(=O)NC(C(C)NC(=O)CCc2nccs2)(C)C)ccc(O)c(C(C)(C)C)c1 c1(OC)ccc(C(=O)NC2CC(C)CN(C(c3nnn(C)c3C)=O)C2)c(F)c1 C(=O)(C1=CCN(C(=O)CC2(C)CCOC2)C1)N(C(c1cccnc1)C)C c1(CN2CCC(CC)C2C(C)C)noc2ccc(OC)cc12 N1(C(CNC(CCC)=O)=O)CCC(N(C(=O)C(C)N(C)C)CCC)CC1 c1(C(=O)NCCCNC(CCCSC)=O)cnc2ncc(Cl)cn12 C(=O)(C(C)P(C)(C)=O)NC(CNC(c1c(C)oc(Cl)n1)=O)C(C)(C)C C1(CC#C)(C(N2CCC(C(C)NC(=O)CSC3CCOC3=O)C2)=O)CCCC1 C#CCCC(O)C(=O)N1CC(CNC(=O)CCC(=O)c2cc(Cl)sc2Cl)C1 C1(NC(C(CC)O)=O)CCc2nc(NC(c3ncn(C(C)C)n3)=O)sc2C1 Cc1[nH]nc(Cl)c1C(=O)NCCCNC(C1(CF)CC(F)(F)C1)=O N1(C(C(CNC(C(COC)(F)F)=O)C)=O)CCC2C(C(N)=O)C2C1 C(CN=c1[nH]c(=NCc2ccc(Cl)cc2)c2sccc2[nH]1)c1nc(C)cc(C)n1 Cc1oc([N+](=O)[O-])cc1C(=O)NC1CCCC(NC(C2(C)CC=CCO2)=O)C1 N1(C(C2C(C(C)O)C2)=O)CC=C(CNC(C2C3CCCC23)=O)CC1 c1(N2CCC(N(CC=C)C)C2)nc2ccsc2c(=NCCN(CC)CCNC)[nH]1 C#CC1CCCC(CN(C(=O)CC(=O)N(C)C)C)C1.C1(=O)CC2(CC2)N1 N1(C(C2CCN(C)C2=O)=O)CCC(NC(=O)CCc2nncs2)C2(CCC2)C1 CCCC(C(=O)N1CCSCC1C(N1CCC(CC(C)C)CC1)=O)NC(N)=O CC1CCN(C(=O)C(N2CCCC2CF)=O)CC1Cc1ccccc1 C=CCC(C)(CC)C(=O)NCCN(C(=O)CCCOc1ccccc1C)C1CC1 C#CC1(C(=O)NCCC2CC(C)(C)CO2)CCN(C(c2cc(CC)n(C)n2)=O)C1 c1(N2CC(NC(Cc3nc(C)sc3)=O)C(F)C2)nc(S(C)(=O)=O)ncc1C Cc1cc(Cl)c(Cl)cc1C(=O)NC1CC(CNC(c2cnc(=N)[nH]c2)=O)C1 c1(OC)ccc(CNC(=O)C(=O)NC23CCCNC2C3)cc1Br c1(N(CC)CC2CCCCN2C(=O)C(C)CC(N)=O)nc2cccnc2s1 CC1CC(C)(C)CCC1NC(=O)NC1CC(C)OC1C C1(NC(c2ccccn2)=O)CN(C(c2c[nH]c(Br)c2)=O)C2(CCCOC2)C1 c1(SCCC(=O)NC2C3CN(C(=O)CC4CCC4)CC23)nccc2ccccc12 Cn1cc(C2=NOC(C(=O)NC(C)CCNC(=O)Cn3ncc(Br)n3)C2)cn1 C(=O)(CC(O)CNC(=O)CCCn1cccn1)NC1(C)CCCC1 N1(C(CC(=O)NCC2CC2)=O)CC2OCCN(C(=O)C(O)CC(F)(F)F)C2C1 N1(C(CC)=O)CCN(C(c2cncc(OC(F)F)c2)=O)CC2CCCCC12 c1(C(=O)NC(C)(CNC(c2cncc(F)c2)=O)CO)cc2n(n1)CCNC2=O C1(O)(CN(C(c2cccc(CC)c2)=O)C)CCN(C(=O)C(C)(C)C(C)O)CC1 C1(NC(CCn2ncc(C)c2)=O)CCSC12CN(C(=O)CC13COC(C)(C1)C3)C2 CCCC(C)(O)C(=O)NC(CNC(=O)C#CC1(C(F)(F)F)CC1)C(C)(C)C CC1CN(C(=O)C(N2CCC(OCC(=O)Nc3cccnc3)C2)=O)CCN1 C1(=O)C2c3ccccc3CN2Cc2ccc(C(F)F)cc21.CCC(CO)N.OC Cc1cc(CN2CCC(CC(N3CCC(CO)C(O)C3)=O)C2)nc(C2CC2)n1 C1(CC(=O)N(C)CC2CC2(C)C)CC2(C1)CN(Cc1ccccc1C(F)(F)F)C2 C(=O)(C1CCCc2ccccc21)NCC12C(CN(C(CCCSC)=O)C1)C2 c1(C(C(=O)NCCN(CC=C)CCC)OCC)ccc(C)cc1 Cc1nc(C)n(CCCC(N2CCC(O)(C(F)(F)F)C2)=O)n1 C1(CCOC)CN(C(=O)Cc2cc(C3CC3)no2)CCN1C(C1C=CCCC1)=O CC1(NC(C2NC(=O)NC2=O)=O)CCN(CC(N2CCCC2)=O)C1.C N1(Cc2scc(CC)n2)CCC2(CCN(C(=O)Cc3ccc(F)cc3)C2)C1 N1(C(C(C)(C)C(F)F)=O)CCN(C(c2nn[nH]c2Cl)=O)CC12CCC2 c1(C2(CNC(N(C3CCOC3)CC)=O)CCOCC2)ccc(F)c(OC)c1 c1(C(=O)NCCN(C(CCN(C)CC)=O)CC)ccn(CC(F)(F)F)n1 c1(C(=O)NC2CCC(NC(C=CC(C)(C)C)=O)C2)nnn2c1CSCC2 c1(N2CCC(CNC(C(C(C)(C)C)=O)=O)C2)ncnc2cc(Br)ccc12 CC(O)CCCN(C(=O)CC1(C)CCN1C(=O)C(C)n1ccnn1)C c1(C(N2CCC(NC(c3c(C)onc3)=O)C(C)C2)=O)cc2ccccc2o1 c1(CC(=O)NCCCC(C)NC(c2cc(F)ccc2F)=O)ccnc(F)c1F C1(C(=O)NC(C)CCNC(=O)CCc2cncc(Br)c2)CC2CCC(C1)O2 S(=O)(=O)(c1cnc(O)c2ccccc12)NCc1cc2c(ccc(OC)c2)n1C N1(C(c2c(C)ccc(O)c2)=O)CCC2(CC1)CN(C(=O)C(C)P(C)(C)=O)C2 N1(C(CNC(C)=O)=O)Cc2nccnc2CC1C(=O)Nc1c(Cl)cnnc1Cl N1(C(=O)NCC2C(CC)C2)CCCCCC1c1ccc(C)o1 c1(OC)ccc(C(Cc2ccc(-c3csc(NC(=O)C(C)OC)n3)s2)OC)cc1 CCC(C)C(CO)NC(C1CN(C(C2CCC(C(=O)OC)CC2)=O)CCN1)=O c1(C(=O)NC2CCCN(C(c3c(C)cns3)=O)C2C)cnc2cc[nH]c2c1 C1(CC)CC(NC(=O)CC2CC(F)CN2C(=O)C(c2cnn(C)c2)=O)CCO1 c1(C(=O)NC(C2(O)CCN(C(=O)CC3(O)CCC3)C2)C)cnc2occc2c1 C#Cc1ccc(C(=O)NCCSCC(=O)NCC2CCCCC2F)nc1 CCC(CC(=O)N(C1CN(C(=O)C(C(C)C)n2cnnn2)C1)CC)C(C)(C)C N1(C(C2(C)C=CCC2)=O)CCCN(C(=O)CC2(O)CCCCCC2)C(CO)C1 c1(C(=O)NCc2nc(CNC(C(CC)C(C)O)=O)sc2)nccc2nn[nH]c12 c1(CC(=O)NC2CCC2NC(=O)CC2CCOC2)coc(-c2ccccc2)n1 CCC(C)CCCCC(=O)N(C(C)CNC(c1cccc(Br)c1N)=O)C N1(C(c2nc(C)[nH]n2)=O)CCC(C2CCCN(C(C3CCCOCC3)=O)C2)CC1 N1(C(CCCC(C)(C)C)=O)CCCC12CCCN(C(C1(C)CCOC1)=O)C2 N1(C(C2(CC#C)CCC2)=O)CCC(CCOC)(NC(C2(C)CNC(=O)C2)=O)CC1 C1(C#N)(C(=O)NC(C)C(C)NC(c2ccc(C(N)=O)cc2)=O)CCCOC1 N1(C(CC2C(C)C2)=O)CC2(CCN(C(=O)Cn3cnc(C(N)=O)n3)CC2)C1 c1(C(=O)NC(C(=O)NCCN(C(=O)CC#N)CC)c2ccco2)ccncc1F C1(C2(N(CCC(=O)N(CCC=C(C)C)C(C)=O)CC(F)F)CC2)CCCO1 N1(C(C2(OC)CCSC2)=O)CC(C2CCN(C(=O)C=CCF)CC2)C1 C(=O)(NNc1ccnc(O)c1)NC(CC)(C)CCC(=O)O C1(C(=O)NC(C2N(C(C=COCC)=O)CCC2)C)CC2(CCOC2)C1 CC1C(C(=O)NC(C)(C(=O)N2CCC2(C)CC(C)(C)C)c2cccs2)CCN1C C1(CC(=O)OC)CCCC(NC(C2(c3ccccc3)CCOC2)=O)C1 CC1=NN(C)C(=O)C1CC(N1CCC(CNC(c2ccc(CO)c(Cl)c2)=O)C1)=O C1(NC(C2CCC(C)(CC)O2)=O)CC2CCC(C1)N2C(C1CC1(C)CC)=O C(=O)(CP(=O)(C(C)C)C(C)C)NC1CCN(C(CCSCC)=O)CCC1CO CCCC(C)CC(=O)N1CCCC1C(C)(C)CNC(C1CC(=O)N1)=O c1(C(N(CCCCC(=O)NC2C(C)C2)C)=O)cccn2cncc12 c1(C(N2C(CNC(C3(CC=C)CC3)=O)C(C)CC2)=O)cccc2nc(C)sc12 N1(C(C2CC(SC)C2)=O)CC2OCC(NC(=O)CCOCC(C)C)C2C1 C=CCC(CNC(=O)C(C)OCCCC)C(=O)N(CC(=O)NC)CCOC C1(F)(c2cn(C(C)CC3CCC4CC34)nn2)CCN(C2(c3ccccc3)CC2)C1 C1(C(=O)NC(C)CN(C)C(c2cc(-c3ccoc3)on2)=O)CC2C=CC1C2 C1(C(N2CCN(C3CN(C(=O)COCCN(C)C)C3)CC2)=O)C(F)(F)C12CCC2 c1(C(N2C(C)(CNC(CS(=O)(=O)NC)=O)CCC2)=O)cccc2c1OC(C)(C)C2 C(CN=[N+]=[N-])(C(=O)NCC(N1CCOCC1)C)NC(CCCCOC)=O C1(C(N2CCC(N(C(c3cn(C4CC4)nn3)=O)CC)C2)=O)CNC(=O)CC1C C(C(C(=O)O)NCC(=O)NC)NC(C(C1CCCC1)NC)=O C1(C(=O)N(CC(C)NC(=O)C(F)CC2CCC2)C)(CC)CCCO1 c1(C(CNC(=O)COC2CCCC2)NC(C(C)O)=O)cccc(Cl)c1 N1(CCC)C(=O)CCC1C(=O)Nc1ccc(-n2cccc2)cc1 c1(C(=O)Nc2nc(C(=O)OCC)c(Cl)[nH]2)cnc(O)c(COC)c1 C(=O)(CC1COc2ccccc21)N1CCC(C)(NC(=O)C=CC2CCCCC2)C1 C1(C#CC(=O)N(C2CCC(CNC(=O)CC(C)n3ccnc3)CC2)C)(CC)CC1 CCCC(CCCNC(=O)C(C)(CC)CO)NC(=O)CCSc1ccccc1F C1(CNC(c2cn(CC)nc2C(F)(F)F)=O)CCCCCN1C(=O)CC(F)(F)F C1(NC(CN(CCC)C)=O)CC(CNC(c2scnc2C)=O)C1(C)C C(=O)(C(C)(O)C(C)C)NCC(C1CCN(C(Cc2nc(C)oc2)=O)CC1)F c1(-n2cc(CSC)nn2)ncc(Cl)cn1.CCC1C(=O)N(CC(=O)O)N1CC(=O)O C1(CNC(=O)CCCF)CCCCCN1C(=O)C=CC1CCCO1 c1(C(N2C(C(=O)NCC)CCC(C)C2)=O)cc(Br)cc(OC)c1OC C(=O)(C(C)(C)C(C)(F)F)N1CCC(O)(CN(C(=O)Cn2cccn2)C)C1 C1(CC(=O)N(CC(C)NC(=O)CC2CCOC2)C)CCCCC1C N1(C(c2ccc(COC)cc2)=O)CC(NC(=O)C(C)(Cl)Cl)CC1(C)COC c1(OC)ccc(CC(N2CC3CC3(CNC(=O)CCC3CNC(=O)N3)C2)=O)nc1 N1(C(C2CC=CC(NC(Cc3c(C)n[nH]c3C)=O)C2)=O)CCc2nn[nH]c2C1 C(=O)(C1=C(Cl)CC1)N(CCC(=O)NCc1noc(C)n1)CC C1(CC=C)(C(=O)NCC(C)(O)CNC(c2cnc(COC)s2)=O)CCCCC1 c1(C(=O)NCCC2CCCN(C(C(CCC)NC(C)=O)=O)C2)ccc2c(c1)CC2 Cc1cc(Br)cc(F)c1Cn1nc(C)c(-c2ccccc2)c1C Cc1cc(C(=O)N(CC(C)NC(C2CCN2C(=O)OC(C)(C)C)=O)C)ncc1F c1(C(=O)NC(C)CC(=O)NCCOc2ccccn2)cc(O)ncn1 c1(CC(N2CC(N(C(C3CC(C)OCC3)=O)C)C2)=O)cccc(F)c1Cl O(NC(=O)CN(C(=O)COCCOC)C1CC1)CC.c12conc1NC2=O N1(CC)CCN(CCc2ccc(NC(=O)C(C)CCCC)cc2)C(C)CC1C C1(NC(C(CCOC)NC(C2CC(C#C)(O)C2)=O)=O)CC(=O)NC(=O)C1 C(CN1C(=O)COc2ccccc21)(C(=O)NC1CCCC1)N1CC2C(CC)(C2)C1 C[Si](C)(C)CCCNC(C1CC(O)CN1C(c1ccccn1)=O)=O CCC(C)(C)CCCC(=O)NCC(O)CNC(C1(CC)CC1(F)F)=O N1(C(C2CC23CCCCC3)=O)CCN(C(=O)Cn2nnc(=O)[nH]2)C2(CCC2)C1 C(=O)(C(F)(F)CC(C)C)NCC(CNC(c1c(C)cc[nH]c1=N)=O)C(F)(F)F N(C1CCCc2n[nH]cc21)C(=O)C(CC1CCC1)NC(C1CC=CC1)=O N1(C(C(C(CC)C)O)=O)CC2CCCC2(CNC(C2CCC(N(C)C)CC2)=O)C1 c1(-c2cnc(CNC(c3ccc([N+](=O)[O-])cc3)=O)nc2)ccc2nccn2c1 C1(CNC(CC(C)(C)O)=O)N(C(=O)CCc2cccc(Cl)c2Cl)CCC1(C)C C(=O)(CCCC(=O)N(C)C)NC(C)CC(C)(C)c1ccccc1 c1(C(=O)NC2CC2SCCO)cccc2nnsc12 Cc1[nH]nc(C(=O)NCC2(NC(=O)CN3CCC(=O)CC3)CC2)c1[N+](=O)[O-] CCC(C)C(CN(C)C)NC(C1CC(O)CN1C(=O)CC1CC2C=CC1C2)=O C(CS(=O)(=O)c1cccc(Br)c1)NC(C(CC=C)C(C)C)=O c1(C2C(CNC(C3(C(C)NC(c4cn(CC)nc4)=O)CC3)=O)C2)ccc(F)cc1 C1(CNC(C(C)Cc2ccccc2)=O)CN(C(=O)C(Cl)=CCl)C(C)(C)C1 C1(F)(CNC(C(COC)OC)=O)CCN(C(=O)CCc2ccccc2F)CC1 c1(CC)ccc(C(=O)NC(C)(CSC)C(=O)NCCc2nc[nH]n2)cn1 N1(C(C=C=C(C)C)=O)CCCC(C(N2CCC(CCO)C2)=O)CC1 C1(CC(=O)NCC(N(C)C(C2C=CCC2)=O)C2CC2)CCCC(=O)C1 Cc1cc(NC2C(C)CN(C(=O)CC3CN(C)C3)CC2C)ncc1[N+](=O)[O-] C1(C(=O)NC(C(=O)NCC(COCC)O)C2CC2)CCCSC1C C1(CCC(=O)N(CC(COC)C)C)CCCCN1C(=O)C=C(C)C(F)F C1(C(=O)NC(CC)(COC)CC)CCCCN(C(=O)CCC2CC(C3CC3)C2)C1 CC1C(NC(c2c[nH]c(=N)nc2C(F)(F)F)=O)CCCN1C(c1cn(C)cn1)=O C1(NC(c2c(SC)csc2)=O)C2CC(O)C1N(C(=O)C1=CCCC1)C2 C(CC1CC1)(C(=O)NCC1(CNC(=O)C(C)CSC)CCCC1)OC C(C(O)C(=O)N1CCC(c2cn(Cc3cc(C4CC4)no3)nn2)C1)OC Cc1ccc(C)c(SCC(N2CCCN(C(C3CC4CC4C3)=O)CC2)=O)c1 c1(SCC)n[nH]c(=NC(=O)N2CCC(c3cn(CCCOCC(C)C)nn3)C2)s1 c1(C(N2CC3C(CNC(c4ccn(CCC)n4)=O)(C3)C2)=O)cc2c[nH]cnc-2n1 Cc1nc(S)sc1CC(=O)NCC1CC(NC(=O)C(C)OCC2CC2)C(O)C1 S(=O)(=O)(c1cc(F)ccc1O)N1CCC(NC(=O)Nc2ccc(C)cc2)C1 C=CCC(C(=O)NCC1CCC(NC(c2cc3cccnn3c2)=O)CC1)C(C)C O=C(C#CC1CCCCO1)NC1(CO)CCN(C(C2CN3CCC2CC3)=O)C1 N1(C(CSCCC#N)=O)CC23CCCC2(C1)CN(C(=O)CC1CC2CC2C1)C3 CC1SCCCC1C(=O)NCCOCC(=O)NCc1ncoc1C1CC1 c1(OC)cccc(C(F)(F)F)c1S(=O)(=O)NC(C#N)C(=O)OC(C)(C)C C1(C(=O)NC(C#C)C(C)OC)C2CC3C(C2NC(C2CC(C(C)C)C2)=O)C13 C1(C(=O)O)(Cc2cn(C3CC(NC(CCCSC)=O)C3)nn2)CCOCC1 CCC(C(=O)N1CCCC1CN(C)C(c1occc1C)=O)c1ccccc1 C1(C(=O)NC(C)CNC(c2ncccc2Br)=O)CCCC12CCC2 C1(NC(C=C(NC(C)=O)C)=O)CC(O)CN(C(c2nc(C)ncc2Cl)=O)C1 c1(C(C(=O)NCCCC2CC2)N(C)CC2(OC)CCOC2)cccc2sccc12 CC1CCCC1NC(C1(CCNC(=O)Cn2nccn2)CC1)=O C1(NC(=O)NCC2N(C(=O)OC(C)(C)C)CCC2(C)C)CCC2C(C1)C2(F)F C(=O)(C(CCNC(=O)CC1CC2(CCC2)C1)OC)NC(C=C)COC c1(CNC(Cc2cccc(C)n2)=O)ccc(C2=CC(=O)CCC2)nn1 C1(CC)CCOCC1(c1nnnn1CCCF)NCCC(C)(C)CO C12(CNC(C(=O)NC3CCC(C)C(C)C3)=O)CCC(CC1)NC2=O Nc1cccc(C(N2CC(CO)C2CC2(C(=O)N)CCCO2)=O)n1 c1(C(=O)NCCCCC2CN(C(CSCCC#N)=O)C2)coc2c1COC2 CCCCC(CC)CC(=O)NC1CC(OC)CN(C(C2CCS(=O)(=O)CC2)=O)C1 N1(C(N2CC(n3cc(CC(c4ccco4)O)nn3)C2)=O)CCCCC1CO C(COC)(CC(=O)N(C(C)CN(C)C)C)NC(c1n(CCC)ncc1)=O c1(C(N2CCC(COC)(NC(=O)CC3CC34CC4)C2)=O)ccc(Cl)c(F)c1 N1(C(C(CC=C)(C)C)=O)CC2CCN(Cc3cc(Br)c(F)cc3O)C2C1 CC1CC(C(=O)N(c2cccc(-c3nn[nH]n3)c2)CC(F)F)C(C)O1 N1(C(c2c(C)noc2C)=O)CCN(C(=O)CC2CC(C3CC3)C2)C(C2CC2)C1 c1(C(N2CCN(Cc3cnc(Cl)cn3)C(C(F)(F)F)C2)=O)ccnc(Br)c1F Cc1cc(CC(N2CCN(C(c3cc(N)ccc3Cl)=O)CC2C)=O)cc(O)n1 c1(NCC(CC(C)(C)C)OC)[nH]c(=NCc2ccccc2SC)nc2scnc12 C1(NC(C2CCCN(CC(C)C)C2)=O)CN(C(C2C(C)C2C)=O)CC1(C)C N1(C(C(=O)N(C)C)=O)CCC2CCN(C(c3nccc4ccncc34)=O)CC12 c1(C(=O)NC2(CNC(C3(C4CC4)CCCO3)=O)CCOC2)cc2ccncc2s1 c1(OC)cc(Cl)c2c(c1)N(C(c1cccc(-c3csc(C)n3)c1)=O)CCC2 C1(C(=O)NCC2(CC(=O)NC(c3ccnc(C)n3)C)CC2)(OC)CCCCC1 c1(OC)cccc(C(C)C(N2CCC(C)C2CNC(=O)Cn2cnnn2)=O)c1 C1(CNC(COCC(=C)C)=O)CN(C(=O)Cc2cnccn2)C2(CCOCC2)C1 C(C1CS(=O)(=O)c2ccccc21)c1n(C(CC)C)nc(-c2ccc(Cl)cn2)n1 c1(CNC(=O)NC2CCN(c3c(OC)cccc3)C2)cc(Cl)cc(Cl)c1OC C1(CC)C(NC(=O)CCOCCSC)CCN1C(=O)C(C)O c1(C(C(N2CCC(CN(C)C(C3(O)CC(C)(C)C3)=O)C2)=O)CO)ccc(Cl)cc1 c1(C(N2CCCC(OC)C2)C(=O)NCC(C)C)cc2ccccc2cn1 C1(C(N(CCC(C)NC(CNC(CC)=O)=O)C)=O)Cc2ccc(F)cc2C(=O)O1 C(=O)(N=c1cc(OC)n(C)[nH]1)C1CCCC(NC(C(CCC)F)=O)C1 CCCCC(F)C(=O)NC(C1CCN(C(c2cc(CC)[nH]n2)=O)C1)(C)C N1(C(c2ccc(C(=C)C)cc2)=O)CCC2(NC(=O)CC(C)(C)C)CCCCCC12 C1(C(=O)NCC2CC=CCC2)CCCCCN1C(c1ncc(F)cc1F)=O c1(C(=O)NCC(C)NC(C(C)OCC2CC2)=O)cccc(C2(C#N)CC2)c1 C1(CN(C(=O)Cc2ccncc2Cl)C)CCCCN1C(c1cnn(C2CC2)c1)=O Cc1ccsc1C1CC1C(N1CC(CO)(NC(=O)Cc2nccn2C)C1)=O N1(C(c2ccc(C)[nH]2)=O)CCOCC(C(=O)N(C)CCC2CCCN2C)C1 C1(NC(CCN(CC)CC)=O)CCC(O)CN(C(C2CCCN(C(C)C)C2)=O)C1 c1(C(=O)NC2C(C(NOCCCCC(=O)OC)=O)COC2)cc(C)nc(C)c1 c1(C(COC)NC(c2conc2C2CC2)=O)ccc(OC(F)F)cc1 c1(N2CC(c3ccccc3)(N(C(=O)CC3CCC(O)C3)C)C2)nc(CO)nc(=N)[nH]1 c1(NC)ccc(C=NOCCC(c2ccc(C(C)C)cc2)(C)C)cc1 c1(CC(=O)NC23C(OC)CC(CC2)C3)c(C)[nH]c2ccnn2c1=O Cc1cn2c(n1)C(C(=O)NCC(CO)NC(=O)C1CC1)CCC2 C(=O)(C(F)C(C)C(F)(F)F)NC(C(C)C)CCNC(=O)C=C1CCC1 N1(C(C23CC(n4cc(-c5c(C)c(F)ccn5)nn4)C2C3)=O)CCC(F)(F)CC1C C1(CNC(c2c(OCC)oc(C)n2)=O)CCN(c2nc(CC)ns2)C12CC2 N1(C(CNC(=O)OC)=O)CC(F)CC1C(N1CCNC(=O)C1)=O C12(CNC(C(C(C)C)NC=O)=O)CCC(CN(C(=O)C(O)C3CCCC3)C1)C2 c1(COC)ccc(C(N2CCCC(C)CC2)C(=O)NC(C)C(=O)OC)c(Br)c1 c1(OC)cc(CNC(=O)C(=O)N(C2CCS(=O)(=O)C2)C)c(OC)cc1Cl C1(NC(c2ccc(N)cn2)=O)CN(C(=O)CCCC2CC2)C2(CCCC2)C1 n1(CCC(N2CCC(NC(c3c(C)occ3)=O)C2(C)C)=O)cc(S(N)(=O)=O)cn1 c1(C(=O)CN(C2CCOC2=O)C2CC2)cccc2ccoc12 C1(N(C(CC2(C=C)CN(C(=O)C(C)(C)N(C)C)C2)=O)C)CCN(C)C(C)C1 CC(=O)CCCC(=O)NCCCCC(C)NC(c1cnnn1-c1ccccc1)=O c1(C(=O)NC2CCCN(C(=O)CCc3cnco3)C2)ccnc2[nH]nnc12 N1(C(C(CCCOC)NC(c2ccc(OC)o2)=O)=O)CC(C)CC(C)(C)C1 C1(C(=O)NCC(CC)(O)CC)CC12CCN(C(=O)CN(C)CCOC)C2 c1(CNCC(c2ccccc2)OC)nc(-c2cnn(C)c2)cs1 C1(NC(CCC2(NC(=O)CCCn3cccc3)CCC2)=O)CC2(C1)CC2(F)F C(C(C(F)(F)F)n1cncn1)NC(c1n(C(C)(C)C)nnn1)C1(CC#N)CC1 C1(F)(C(N2CC(C(=O)NCC(C)(C)n3cccn3)C(F)C2)=O)CCCCCC1 C(=O)(CCC(C)C(C(=O)NCCC1CC1)N1CCC(OCC(N)=O)C1)OC N1(C(C(C)C2CCC2)=O)CC2COCC(C1)C2NC(c1cn(C2CC2)nn1)=O c1(C(N(CCCNC(CCOCCOC)=O)CCO)=O)c[nH]nc1F C=CCC(CC)C(=O)NC(CCC)CC(=O)NCc1cn(CC)nn1 N1(C(COCc2cc(C)on2)=O)CCCC2CCN(C(=O)C=CC3CCC3)CC12 C1(CCC)CN(C(C2COCCN2C)=O)CCN1C(C1CC(F)(F)C1)=O c1(C(=O)NC(CC)CN(C(=O)C(c2ccc(Cl)s2)C)CC)cc(C#N)c(C)cn1 C1(C(=O)NC(c2nc(NC)sc2)C)CCCN2CCCCC12 C(CC(C(C)C)NC(=O)C(C1CCN(C(=O)CC2(OC)CCCCC2)C1)F)OC c1(OCC)ccccc1CCC(=O)N(C(C)CCNC(=O)CP(C)(C)=O)C Cc1cc(C2CC2)oc1C(=O)NC1(C2CCCN2C(C2CCC3(CC3)C2)=O)CC1 C1(N=[N+]=[N-])(C(N(CCN(C)C)CC)=O)CCN(C(=O)CC2CCCCO2)C1 CCCCCC(C)CC(=O)N1CCC1CC(=O)NCC1(CO)CCCO1 CC1CN(C(=O)CCCCn2ccnn2)CC1(C)CNC(C1CCS(=O)(=O)C1)=O CC(CC(=O)NCC1CC1CNC(C1(F)CCC1)=O)C1CC1 c1(C(=O)NCCCCC(=O)NC2CCC(C)NC2=O)ccc2cccnn12 C=CC(C)(C)CC(=O)NCC1CC(NC(=O)CCNc2ccccn2)C1(C)C c1(CC(C)C(=O)N2CCCC2CN(C)C(C2(C)CC2)=O)ccc(F)cc1F C1(F)(CNC(C2CC=CC2)=O)CCN(C(C2CCC(F)(F)C2)=O)CC1 CCC1=NOC(C(N2CC(O)(CCNC(C3CCOC(C(C)C)C3)=O)C2)=O)C1 c1(OC)cc(CN2CC=CC2C(N2CCCCC2CCO)=O)cc(Br)c1O C1(C(N2C(CNC(C(C)C(F)F)=O)CN(C)CC2)=O)C2CC3CC(C2)CC1C3 N1(C(C(C)C(C)(C)C)=O)CCC(C2(O)CCN(C(C3COC(=O)N3)=O)CC2)CC1 Cc1ccnc(C)c1C(=O)NC1CCCN(C(=O)Cn2cc(C(C)O)nn2)C1C C(=O)(C1CCCc2n[nH]cc21)NC1C=CCN(C(c2nc(C)nc(O)c2)=O)C1 CCC(C)(C)C(O)C(=O)N1CCN(C(c2ccoc2C)=O)C2CCC12 c1(C(N2C(C)CC(CNC(C(CC)F)=O)C2)=O)ccc(F)c(OC)c1 c1(C(=O)NCC2CCN(C(c3cc(C(N)=O)oc3)=O)C2)cc(Cl)c(Br)[nH]1 CCC(C)CC(=O)NC(CN(C)C)C(=O)NCCC(=O)OCCOC C(=O)(C1=NOC(C)C1)NC(C1CCN(C(Cc2n[nH]c(=NC)s2)=O)CC1)(C)C c1(C(=O)NC2C(NC(CCC(C)C)=O)CC2)n[nH]c2ccc(O)cc12 c1(C(C(=O)NC2C(CNC(C3(C(=O)OC)CC3)=O)C2)C)cn(C)nc1C CCCC(F)(F)C(=O)N1CC(N(C(=O)CC2CCCCCC2)C)C1 N1(Cc2c(C)cns2)CCCCC1C(C)N CC(C)(C(=O)NCCNC1CCC(c2ccccc2)OC1)S(C)(=O)=O C(N=c1[nH]c2cccc(Br)c2o1)C1(C)CCC(NC(C2(CC)COC2)=O)CC1 c1(-n2c(C3CC3)nc(C(C)C)n2)ccc(S(=O)(=O)NC2CCCS2(=O)=O)cc1 c1(C(=O)NC(C(C)O)C(=O)NCCc2ccccn2)ccn2cncc2c1 C1(NC(CCCCOC)=O)CCC2(CC1)CN(C(c1cc[nH]c(=N)c1)=O)CCO2 N1(C(C2(C(=O)OCC)CCO2)=O)CCC(C)C(NC(=O)C(C(C)(C)C)SC)C1 C1(F)(C(=O)NC2CCN(C(CN3C(C)CCC3)=O)CC2)CC2(CCC2)C1 C1(O)(C(CC)C(=O)NCC2(OC)CN(C(c3cnc(S)[nH]3)=O)C2)CCCCC1 CC1(CNC(c2ccc(CO)s2)=O)CCN(C(C2(c3nccs3)CC2)=O)C1 C1(CC(N2C(CNC(c3ccc(OC)o3)=O)CC(O)C2)=O)CCCCCCC1 C(C)(C(=O)N(CCC(C)NC(=O)Cc1ccccc1Cl)C)(C(C)C)OC c1(COC)ccc2ccc(-c3nc(C4CC4)nn3-c3ccc(Br)c(Cl)c3)cc2c1 c1(C(=O)NC2CCC(NC(c3cn(CC=C)nc3)=O)C2)cc(C#N)cc(C)n1 CCC(C)C(C)NC(=O)CCOCCNC(=O)CCc1cnc(C)o1 N1(C(c2c(C)nc(C)[nH]2)=O)CC2CC(NC(=O)Cn3cc(Br)c(C)n3)C1C2 c1(C(N2CC(NC(c3ccc(C)nn3)=O)C(CO)CC2)=O)c(C)cc(C)nc1O C(CSC)(C(=O)NCC(C1CCC1)NC(c1sccc1C)=O)OC C(C(=O)NNc1cc(Cl)ccc1[N+](=O)[O-])(c1cccnc1)N(C)C C(CCCC#N)(C(=O)NC(c1cccc(F)c1)C1CCOC1)N(CC)CC1CCC1 CC(=O)CCCC(C)C(=O)NC1(C(=O)NC2(CC3CCC3)CC2)CC1(C)C CCCC(CCC)CC(=O)NCCn1cc(C(=O)NC2CCN(CCC)C2)nn1 c1(OC)cc(F)c(C(N2CCC(NC(=O)C3=C(C)OCC3)C(O)C2)=O)cc1OC c1(C(N2CC(NC(CN(S(C)(=O)=O)C)=O)C(CO)CC2)=O)cc2ccccc2s1 c1(C(N2CC(C(C)NC(=O)C(CO)NC(N)=O)OCC2)=O)ccc(P(C)(C)=O)s1 c1(C(=O)NCC23C(CN(C(C=Cc4n(CC)ccn4)=O)C2)C3)c(C)ccnc1C CC(CO)CCNC(=O)CC1CCCN1C(=O)C1CC1 c1(SC)ccc(C)c(C(=O)NC(CCNC(c2cnn[nH]2)=O)C(C)C)c1 CC1(C)CC(C(N2CC(n3cccn3)C2)=O)CN(C(c2cc(N)ccn2)=O)C1 N1(C(C=C(C)Cl)=O)CC2(CCC2NC(C2CC(=O)NC(=O)N2)=O)C1 N1(C(c2c(C)n(C(C)C)nc2)=O)CC2CC1CN2C(c1ccnnc1S)=O C1(NC(CCCc2ccc(C#C)cc2)=O)(CO)CC2(CCCCC2)C1 N1(C(c2c(CC)nc[nH]2)=O)CCC(N(CC(C)C)C(c2cc[nH]c2CC)=O)CC1 c1(C(N(CCF)CC)=O)[nH]c2cc(OC)ccc2c1C N1(C(C2(C=C)CCC2)=O)CCC(NC(c2c(F)cccc2F)=O)C(C(C)C)C1 CC1(C)C(C)(C(=O)NCC(C2CCC2)NC(c2cc(N)nc(Cl)c2)=O)C1(C)C N1(C(C(C)Oc2ccccc2)=O)CC(NC(C23CC(C2)C(C)O3)=O)C(C)(C)C1 N1(C(C(C)OCCOC)=O)CC(CC2(CC(=O)N(C)NC(C)=O)CC2)C2(CC2)C1 N1(C(c2c(Cl)ncc(N)c2)=O)CC(CNC(c2nocc2Cl)=O)OC2COCC12 c1(NC2CCCCN(C(C3CN(CCC)C(=O)C3)=O)C2)ncnc2sccc12 C1(CNC(c2ccc(C)s2)=O)CCCN(C(=O)C(CCN(C)C)N(C)C)CC1 Nc1sc2ccccc2c1C(=O)NCCCN(CCO)C(C1CCNC1=O)=O c1(CC(=O)NCC2C(CN(C(=O)Cc3cc(Br)cs3)C)C2)cn(C)nn1 N1(C(c2ncnc(C)c2C)=O)C2CCC1CC(N(C(=O)CC(C)C(F)(F)F)C)C2 C(=O)(C(C)(C)CO)NCCOCCCN(C(=O)Cc1nccn1C)C c1(C(=O)NCCCCNC(C2C(C)CC2)=O)ccnc(C2CC2)n1 CCCCC(CC)C(=O)N(C1CCN(C(=O)CC2CC(=O)C2)C1)CC C1(NC(C=CC(C)C)=O)CC2CCC1N(C(c1cc(F)n[nH]1)=O)C2 C(c1sc(Cl)nc1Cl)=CC(=O)NC1C(CNC(C(COC)OC)=O)C1 C1(C)(C(=O)NC(C)CCN(C)C(c2ccc(Cl)nc2O)=O)CC(C(C)(C)C)=NO1 N1(C(C(CC)CN(C)C)=O)CCOCCC1C(N1CCOC(C)(C(C)C)C1)=O c1(CNC(C2(C)CC2)=O)ccnc(N2CCNCC2)c1.c1(C=O)cnc(S)[nH]1 C(=O)(CCCC(C)NC(=O)CNC(=O)C(C)(C)C)N1CCC(OC)C1 C(=O)(CCN(OC)C(=O)C1(F)CC1)NCC1(CO)C(C=C)C1 C12(C(=O)NC(CC#C)CC(F)F)CCC(CC1)N(C(=O)CC1CCCCO1)C2 c1(C(=O)NCCC(C)NC(C2(F)CCOCC2)=O)ccc2c(c1)CCCS2 N1(CC=CC(=O)NCC2CC(CNC(c3cc(O)ncn3)=O)C2)CCOCC1=O C1(CNC(C2CC(CCNC(c3oc(C)c(CO)c3)=O)C2)=O)CC2CCC1CC2 CC1CCC(NC(=O)C(F)(F)c2cncs2)CN1c1nc(CC2CC2)ns1 C1(NC(CCN(CC)CC)=O)CC2CCC1CN2C(=O)C(O)c1ccco1 CCCC(C(=O)N1CCC(CC(=O)NC(C)C(N)=O)C1)C(C)C c1(C(N2CC(N)(CC)C2)=O)c(C)ccc2cccnc12 C(=O)(CS(=O)(=O)C(C)C)NCCCCC1CN(C(C(C2CCCC2)OC)=O)C1 C1(NC(c2n(C(C)C)ncc2)=O)CC2CCC1N2C(=O)C=Cc1ccc(F)cc1 c1(C(N(C)CC2CCCN2C)=O)cn2c(n1)CCN(C(C1CCC(O)C1)=O)CC2 c1(C(N2CCCC2)CNC(=O)CC2(C3CC3)CC2)cccc(F)c1 C1(NC(C=CCOC)=O)CC2CCC(C1C)N2C(=O)C(c1ccnn1C)C Cc1ccc(C(=O)N(C(C)CCNC(c2nnsc2C(F)F)=O)C)o1 C(=O)(C1=CC2C=CC1C2)N1C(C)C(C(=O)NCC2CC3CCC3C2)CC1 N1(C(c2cc(C(CC)C)no2)=O)CCC(NC(=O)CCSCC(N)=O)C1C(C)C c1(-n2ccc(CNC(C(=O)NCC)C)n2)cccc(Cl)c1 Cc1cc(Br)cc2[nH]c(C(N3CC(CN=c4[nH]ccnc4F)C(C)C3)=O)cc12 C=CC1(NC(=O)CC(C)(C)NC(c2ncsc2NC)=O)CCCC1 c1(NCCCC)[nH]c(=NC2CC2C)nc2c1cnn2C Cc1ccc(O)c(CNC(=O)CC(CC2CC2)NC(=O)C(N)=O)c1 N1(C(C(C)c2cccs2)=O)CC2(C(=O)NC(CO)CCC3CC3)CC1CCO2 C1(C(=O)NCCS(=O)(=O)NC(=O)CSCCC(C)C)(SC)CCCC1C C(=O)(CCS(=O)(=O)Cc1ccccc1)NC(C)CC1CN(C(=O)C(Cl)=CCl)C1 N1(C(=O)CCc2cn(-c3cccc(Br)c3)nn2)CCC(O)(CN2CCCC2)CC1 C1(C(=O)NC2C=CCC2)CCCN(C(C2CCCC2)=O)CC1 N1(C(c2c(OC)nsc2)=O)CC2(NC(c3coc(Cl)n3)=O)CC1C2 N1(C(C2(OCC)CCCC2)=O)CCC(CC(C)NC(C2(CC)CCC2)=O)CC1 C1(CNC(=O)C=CC=C(Cl)Cl)CC2(CC2)CN1C(=O)CC1CC(C(F)F)C1 CCCCC(CC)C(=O)NC(CCCNC(=O)C=C(C)C(C)C)c1ccccc1 C(=O)(C#CC1CCCCC1)NC1(COC)CCN(C(=O)CNC=O)C1 c1(C(=O)NC(C2CCCO2)CO)ncccc1OC(F)(F)C(F)Br N1(C(CC2CC(C)(C)C2)=O)CCN(C(c2cccc(C(=O)OC)c2)=O)CC1 CC(C)CC(C)(C(N)=O)NC(C1CC(NC(c2ccnc(CO)n2)=O)C(O)C1)=O Cc1ccc2c(n1)N(C(=O)C(N1CCc3ccccc3C1)=O)CCC2 c1(OC)cc(OC(c2ccc(C(F)(F)F)cc2)=O)c(Cl)cc1C#N c1(CNC(N2CCN(C3CC3)C(=O)C2)=O)nc2cccnc2[nH]1 c1(NC(C2CCC(NC(C3CC4CCC3O4)=O)C2)=O)cccn2ncnc12 C12(CNC(C3CC4C=CC3C43CC3)=O)CCC(CN(C(c3cccnn3)=O)C1)C2 Cc1[nH]c(C(N2CCC(C)C(NC(=O)CS(=O)(=O)CC)C2)=O)c(C)c1C N1(C(COCCC#C)=O)CCC(CNC(c2ccn(C(C)(C)C)c2)=O)C1 O=C(C1=COCCO1)NCCC1CC(NC(C2(F)CCOC2C)=O)C1 C1(NC(COc2cccc(OC)c2)=O)CCN(C(=O)C=CC(C)C)CC1O CC(Cc1ccco1)N=c1cccc(S(=O)(=O)NCCc2cnco2)[nH]1 CN1CCC(N(C)Cc2c(Br)nnn2C)C1=O c1(C(=O)OC)ccc2c(c1)CCCN2C(=O)NCc1ncc(C(F)(F)F)[nH]1 C1(NC(=O)CC2C=CCCC2)CCCCN(C(=O)C(O)CN2CCOCC2)C1 C1(N(C(CNC(CNC(C)=O)=O)=O)C)CN(C(=O)CCCC(N)=O)CCC1C CN1CC2(CCCN(C(CCCC3CC3)C(=O)NC(C)(C)C)C2)CC1=O C(=O)(CCCC(C)(F)F)N(C)CCN(C)C(C1(COC)CCCO1)=O.C1(CC)CC1 C(CC(C)(C)C(=O)NC1CCCC1CNC(=O)CC1CCC(=O)NC1=O)SC c1(OC)ccc(C)nc1C(N1CCC(N(C(=O)C(C)n2ccnn2)C)CC1)=O C(=O)(C(C1=CCCCCC1)N1CC(C)(C)CC1C)NC(C(=O)OC)C c1(CC)noc2ncc(C(N3CC(NC(=O)CCF)CC(O)C3)=O)cc12 CCCC(C(=O)N1CC(F)CC1C(N1CCCC(CC2CC2)C1)=O)n1cccc1 C1(C(=O)NCC(F)CO)(SC)CN(C(=O)Cn2ccc(C)n2)C1 c1(C(=O)NCC2(NC(CC(C)O)=O)CC2)cccc(Cl)c1O Cc1cc(=NC(=O)C2CCN(C(c3ccn(C(F)F)n3)=O)CC2O)[nH]n1C c1(CC(=O)NC(C2CCCCC2)CNC(C(CC)SC)=O)c(F)cccc1F c1(C(C)NC(N2CC[Si](C)(C)C2)=O)ccc(F)c(F)c1 C1(C)(C(=O)NC2C(OC)CN(C(=O)CCCCSC)C2)COCC1(F)F C(=O)(C(F)(F)CC(C)C)NCC1(C)CCCN(C(C2(CC#C)CC=CCC2)=O)C1 N1(C(C2(CC)CC(C)(C)C2)=O)CCC(NC(c2cnc(N)c(Cl)c2)=O)C(CO)C1 CC#CCCCC(=O)N1CCCC(C(C)NC(c2ccc(C)nc2)=O)C1 C(=O)(C1=NOC2(CCC2)C1)N1CC(C)C(NC(c2cnc(O)n2C)=O)CC1 NC(Cc1ccc(F)cc1)CC(=O)N1CCNC(c2cccc(Br)c2)C1 c1(C(N2CC(NC(c3nccc(C)n3)=O)C3(C2)CC3)=O)ccnc2[nH]c(C)nc12 CC(C(=O)NC1CCCCC1NC(c1cncnc1)=O)S(=O)(=O)C1CCOCC1 Cc1c(-c2ccc(C(=O)Nc3nc(Br)ccc3O)nc2)ccnc1F CC1(CNC(=O)CC2CCC2)CN(C(=O)CC2CCCC2)CCO1 C1(C(=O)NCC(CNC(CC2(C)CC2)=O)C(F)(F)F)CCn2ncnc2C1 C#CC1(C(N2CCC2(C)CC(=O)NCc2ccc(C)s2)=O)CCCCC1 N1(C(c2cccc(C(N)=O)c2)=O)CCC2(CCN(S(=O)(=O)CCBr)C2)C1 c1(C(=O)NC2CC(NC(C3CC(C)OCC3)=O)C2)cnc2n1CCOC2 c1(C(=O)NCC(CNC(c2c(CC)noc2C)=O)C)c[nH]c2cc(Cl)ccc12 N1(C(=O)NCC2C(C)COC2)CCSCCC1C c1(C(N2CC(NC(=O)CN3Cc4cncnc4C3)C2)=O)ncc2nc(Cl)nc-2[nH]1 CC1Cc2c(N)cccc2CN1C(=O)NC1CC2(C1)CC(O)C2 N1(C(Cc2c(C(C)C)con2)=O)CC(N(C(=O)Cc2ncc(F)cn2)C)C(O)C1 CC1(C)C(NC(=O)CC2CC(F)C2)C2CCCN(C(C3COC4COCC34)=O)C12 N1(C(C2N(C(CC(C=C)C)=O)CC=C2)=O)Cc2cccc(C#N)c2C1 c1(C(N(CC(C)N(C)C(c2cnns2)=O)C)=O)cccc(C2CC(F)(F)C2)c1 N1(C(c2n(CC#C)ccc2)=O)CC(NC(C2CC(C)(C)C2)=O)C(CC2CC2)C1 c1(CC)ccc(C(C)C(N2CCC(C)(NC(=O)CS(=O)(=O)NC3CC3)C2)=O)cc1 C(CN=c1nc(C(F)(F)F)cc(C(F)(F)F)[nH]1)c1cc(C)nn1C C1(CC(=O)N(CCCNC(C(CC)CC)=O)CC2CCCC2)CCCNC(=O)C1 c1(-n2ccc(C(N3CC(NC(C(C)(C)O)=O)C(F)C3)=O)n2)ccc(F)c(F)c1 C1(NC(C(COC)C)=O)CCCCC1NC(C1CC(N2CCCC2)C1)=O c1(CC(N2CC(N(C(=O)CC3CCOCC3)C)C(O)C2)=O)ccc2ccoc2c1 c1(C(N(CC(CC)NC(=O)CC2(C(F)F)CC2)CC)=O)cc(CO)ccn1 c1(C(N(C2CN(C(C(=O)Nc3ccc(C)cc3)=O)C2)C)=O)ccnc2cc[nH]c12 C1(C)(NC(c2c(COC)cco2)=O)CCCCC1C(=O)N(C1CCC1O)C N1(CC(=O)NCc2c(C)cncc2)CC2CCC1CN2C(c1cccc(C)c1)=O C12(C(=O)NC(c3ncc(C)[nH]3)CC)COCC1CN(C(C1CCCC(CF)C1)=O)C2 c1(C(N2CCN(C(c3cn(C4CC4)cn3)=O)CC2)=O)cnc2ccc(F)cc2c1 C1(C2(O)CCOCC2)(CNC(c2nccc3nn[nH]c23)=O)CC1 c1(C(N2C(C3(C(=O)NCC(COC)OC)CC3)CCC2)=O)nccc(C)c1N n1(C(C(=O)NC(CC)CNC(c2cc3sccc3[nH]2)=O)C)cnc2ccccc12 Cc1cc(C(=O)N(C(C)CCNC(C2(CC(F)(F)F)CC2)=O)C)c(C)[nH]1 C1(n2cc(CN3CCC(C(C)=O)C3)nn2)CCN(C(=O)CCS(C)=O)CC1 Cc1ccc(CCN2CCCC(C(=O)N(C)CCO)C2)cc1 C1(C(N(CC(C2CCC2)OC)C)=O)CCC2(CC2)N1C(c1csnc1Cl)=O CCC(C)C(C)C(=O)N1CCC(C)C(NC(c2cccn(O)c2=O)=O)C1 N1(C(C(COC)COC)=O)CCN(C(c2ncc(Cl)cc2O)=O)CC1CO C1(NC(C(C)SCCCC)=O)CN(C(c2nnn(C)c2C)=O)CCC1(C)C N1(C(c2ccn(CCC)n2)=O)CCCC(O)(CNC(c2ccc(C)c(N)c2)=O)C1 N1(C(Cc2ccc(C)cc2C)=O)CC2(CCCC2CC(N2CCNC(=O)C2C)=O)C1 c1(C(=O)Nc2ccc(NC(C)=O)cc2F)cc(Cl)c(F)cc1O C1(CNC(C2C3COCC23)=O)CCC(C(N2CCCC(CC3CC3)C2)=O)CC1 c1(C(=O)NC2C(NC(C(C)CS(C)=O)=O)C2)cc([N+](=O)[O-])ccc1O Cc1nn(-c2ccc(Cl)cc2)c(Cl)c1CNCc1cnc(CN2CCOCC2)s1 n1(C(C(=O)NCCOCCCN(C(C(C)CC2CC2)=O)C)C)cnc(C#N)n1 CCC1=C(C(=O)NCC2CC3CCC2N(C(C2CN(C)C2)=O)C3)SCCO1 c1(C(N2CCCC(CNC(C(C=C)(C)C)=O)C2)=O)c(C)nn(CC)c1Cl CCCCCCCCC(=O)NC(CC(C)(C)C)C(=O)Nc1cccc([N+](=O)[O-])c1 c1(-c2cc(C(N(OC)C)=O)cc(F)c2)cc(C(=O)NC2CC2(F)F)cc2[nH]ncc12 CCCCCCC(C)C(=O)NCC#CCNC(=O)C(CC)OC(C)=O c1(C(N2CCSC(C)C2)C(=O)NCC(=C)C)ccc2c(c1)CCCS2(=O)=O CCCC(O)C(C(=O)O)NC(C1CCC(NC)CC1)=O c1(C(=O)NC(C2CN(C(c3cc(COC)on3)=O)C2)C)ccc(F)c(C)c1Cl c1(CC2C(=O)N2)ccc(Cl)cc1Cl.N1(C(C(C)SC)=O)CC(O)CC1C(C)C C(C(=O)N1CC(O)C(O)CO1)c1ccc(C(N2CC(C)OCC2C)=O)cc1 CCCCCCN(C(=O)CCN(C(C1COC(C)C1)=O)CC)CCO C(=O)(C(C)C(C)COC)NC(CC(C)NC(CCc1ccc(OC)cc1)=O)C N1(C(CC2CCCC(C)C2)=O)CCC2(CCN(C(=O)Cc3cnoc3)CC2)C1 N1(C(c2cc(CC)n(C)n2)=O)CCN(C(c2nccc(C(F)(F)F)n2)=O)C(C)C1 C1(NC(=O)C=C2CCOCC2)CCCC(CNC(=O)CCn2cnnn2)C1 CP(C)(=O)CC(=O)N1CC(C(N)=O)(CNC(c2ccc(CN3CCCC3)o2)=O)C1 c1(C(=O)NC2C(CNC(COCP(C)(C)=O)=O)C2)ccc2n[nH]cc2n1 c1(CC)ccccc1-n1cc(C2C(C)CCN2C(=O)CCC(C)N(C)C)nn1 C12(C(N3C(CN(C(c4cc(C)oc4)=O)C)CCC3)=O)CCCC1(C(N)=O)C2 N1(C(CCn2c(C)ncc2)=O)CCCC(C(N2CCC(C)C2)=O)C1 N1(C(C(CC#C)C2CC2)=O)CC(CO)C2(C1)CN(C(=O)Cc1ccco1)C2 CC1(NC(=O)CCCC2CCOCC2)CCC(C(F)(F)F)CC1 c1(C(N2CCN(C(c3c(C)nco3)=O)C(C)C2)=O)ncc2[nH]ncc2n1 CC1(C)CC(CNC(=O)CN2CCCCC2)N(C(c2ccc(F)c(Cl)n2)=O)C1 c1(-c2cn(CC(=O)NCC(C3CCCCC3)(C)C)nn2)ccc(Cl)cn1 C1(C(=O)NCCCC(C)NC(C(CC)(C)CO)=O)CCC([N+](=O)[O-])CC1 Cc1nc(CS(=O)Cc2cn(CC3=CCCC3)nn2)no1 Cc1[nH]nc2ccc(C(=O)NC(C3CCN(C(c4cc(N)ccn4)=O)C3)C)cc12 c1(C(=O)NCC2CC2)ccc(OC2CC2)nc1.Cc1ncc(N)o1.C1CC(C)C(=O)N1 N1(C(C2CCCC2NC(C(C)(C)C)=O)=O)CCN(c2cc(F)ncn2)CC(O)C1 C=CC1(CC(=O)NC(C)(CNC(c2ccc[nH]2)=O)C2CCC2)CCC1 N1(C(c2nnn(C(C)(C)C)n2)=O)CCCCC12CNC2 O=C(C#CC1CC1)NC1CCCCC1NC(=O)CC1CCS(=O)(=O)C1 c1(OC)nc(C(=O)NC2CCC2C(=O)NC(c2ccsc2)C)co1 C(C(=O)NC(CC(=O)NC(C)CC(=O)N(C)C)C(C)C)(C(C)(C)C)SC C1(C(=O)NC2OCCN(C(COCC)=O)C2)CCN(c2ncc(C(=O)O)s2)CC1 C1(C(=O)NC)CN(C(=O)Cc2cccc(F)c2)C2(CCC2)C1 C12(CCNC(=O)CC3CCC4CC34)CC3CC(CC(C3)C1)C2 CCC(CC(=O)N1CCOCC1CNC(c1cccnc1O)=O)C(C)C C1(C(N2CCOC3CC23)=O)CCN(Cc2ccc(SC(F)(F)F)cc2)CC1O C12(C(=O)NC(CC#C)C)CC1CN(C(=O)CN(C)C)C2 C(=O)(CS(=O)(=O)C(C)(C)C)NCC1(O)CCN(C(Cc2cc(C)sc2)=O)C1 C1(C(=O)NC(C(=O)N(CCS(C)(=O)=O)C)C2(C)CC2)CCCC(=O)N1C CCCC(C)CC(=O)NC1(C)CCN(C(=O)CC2(C)CCCCC2)C1 C1(C(N2CC3(CN(C(c4nn(CC)c(C)c4)=O)C3)C2)=O)CCOCC12CCC2 C1(NC(C=CSC)=O)CCCC12CCN(C(c1cc(F)cc(C)c1N)=O)CC2 c1(C(=O)NCC2(OC)CCN(C(c3c(C)cnn3C)=O)C2)ccc(S(C)=O)cc1 c1(CC(=O)NCC2CCC(NC(c3ccc(C)s3)=O)C2)ccc(O)cc1Cl c1(CC(C(=O)NC(C(=O)OC)C2CCC2)OC)ccc(OC)cc1 c1(CC)cccc(C(=O)NCC2CN(C(=O)C(C)Cc3cnco3)CCO2)c1 c1(C(=O)NC(CCNC(C(C2CC(F)(F)C2)OCC)=O)C)cc(Cl)ccc1C N1(c2nc(Cl)nc(CC)c2Cl)CC23CCCC2(CN(C(C2CC(C)=NO2)=O)C3)C1 c1(C(=O)NCC2CC(C)N(C(c3ncc(F)cc3F)=O)C2)ccc(F)c(O)c1 C1(C(=O)NC2(CC=C)CCN(C(c3cccn3C)=O)C2)C2CCC1(C)C2(C)C C(=O)(C(C)(CC)C(=O)N1CCCC(N(C)C(c2ccnc(OC)n2)=O)C1)OCC C1(c2nnnn2CC2CCCO2)(NCC(NOCC)=O)CCC2(CC1)CSC2 N1(C(C(C)N(C(C2(C)CCCC2O)=O)C2CC2)=O)CC(CO)CC(C)(C)C1 C(=O)(CC(C)(C)CNC(c1cc(CCO)on1)=O)NC(CN(C)C)CO N1(C(Cc2cccc(OC)c2F)=O)CC(NC(=O)CSCC(C)C)CC2(CC2)C1 C(N=c1ccc(C#N)c(C)[nH]1)C12OCC(CNC(C(C)(C)N(C)C)=O)(C1)C2 C(=O)(C(F)CC(C)(C)NC(C1OCC2CCCC12)=O)NC(c1cccs1)C C(=O)(C(O)CC(F)(F)F)NCC1(C(=O)NC2CC(C)C2)CCCC1 C1(C(=O)NC2(CN(C(C3C(=C)C3)=O)C)CC2)CCCN1C(C)C C1(CNC(C(C)OCC)=O)CC2(CCN(C(=O)C(C)(O)C3CCC3)CC2)C1 C1(CNC(C(C)NC(c2ccoc2)=O)=O)(CO)CCN(C(=O)CC23CC(C2)C3)C1 N1(C(c2c(C)occ2)=O)CCN(C(C2COCC2(C)C)=O)C(CO)C1 c1(C(=O)NCC#CCNC(CC2CC(C)(C)OC2)=O)c(Br)ccc(F)c1N C1(CNC(=O)CCCc2ccsc2)CC2CCC(C1)N2C(=O)Cn1cccn1 CC1(C)CCC(C(=O)Nc2cc(O)cc(F)c2)CN1C(C1CC2(CC2)CO1)=O C1=CC(=O)OC(=O)c2ccc1o2.C(=O)(C(C)N(C)CCC(=O)O)NC(CC)C C1(CC=C)(NC(=O)CC(=O)NC)CC2CCC(C1)N2C(=O)C(O)C1CCCC1 c1(OC)cnc2[nH]c(C(=O)NC3(CO)CCN(C(c4nncs4)=O)CC3)cc2c1 Cn1cc(CCNC(=O)CC2CCN2C(C2CC(F)(CF)C2)=O)nn1 C1(C(=O)NCC(C)(C)N(C(=O)CCSCC(N)=O)C)CC=CCC1 CC1(C)CC(C(=O)NCc2ccc(C#N)cc2)N(C(c2cc(C(F)F)[nH]n2)=O)C1 CC1(C(=O)OCc2ccc(C(F)(F)F)s2)CCc2ccccc21 C1(C(N2CC3C(CNC(CSCC)=O)C3C2)=O)(COC)CCCNS1(=O)=O N1(C(C(C)SCCCC)=O)CCCN(C(c2ncn(C)c2C)=O)CCC1 C1(CNC(C2(CC)CC2)=O)CCC2(CN(C(c3ncc(F)cc3N)=O)C2)O1 n1(CC=C)cc(CC2CCCN2C(c2cc(CCC)[nH]n2)=O)nn1 C(=O)(CCC(C)(C)[N+](=O)[O-])N(C(CNC(C(C(=O)OC)(C)F)=O)C1CC1)C N(C(=NCCC1CCOC1)NCc1ccccc1Cl)CC1CCN(C(C)(C)C)C1 C1(CC(=O)NC2(CN(C)C(C3CC(=O)N(CC4CC4)C3)=O)CC2)CCCCC(=O)N1 c1(C(=O)NCCCC(=O)NC2CCCCCC2O)ccc2[nH]ncc2c1 c1(C(=O)NCC2C(C(N(C)Cc3cnn[nH]3)=O)CCC2)ccncc1Cl C1(NC(c2coc(O)n2)=O)CC(NC(C2CN3CCC2CC3)=O)C12CCC2 c1(SCC(=O)NC(CC)CN(C(=O)C(C)c2ncco2)C)cccc(Cl)c1 c1(CNC(c2ccc(C)cc2)CC)ccc(-c2cnn(C(C)C)c2)cc1F CC1=C(C(=O)N2CCN(C(c3cc(C(N)=O)no3)=O)CC2CF)S(=O)(=O)CCO1 Cc1c(CC(=O)NC(C)(C)CNC(=O)C2=NN(C)C(=O)CC2)oc2ccccc12 C(C)(CCCCNC(=O)CNc1ccc(C(N)=O)cc1)NC(C1C(C)=C1)=O CCC(CCC(=O)NCC1CC1CC(=O)NCc1nc(C2CC2)no1)OC c1(C(=O)NCCCN(C)C(C2(F)CC=CC2)=O)cccc(SCC#N)c1 N1(C(c2cc(OC)ncc2Br)C(=O)NC2COC2)CCC(O)(C#CBr)CC1 C1(NC(c2cc(COC)on2)=O)CN(C(=O)CSc2nncs2)CC2CC12 c1(C(=O)NC(C2CCCN2C(=O)CN2CCOCC2)C)cccnc1S Cc1csc2ccc(C(=O)Nc3ccnn3C3CCOC3)cc12 c1(CC(N2C(C)(C)C(CNC(C3CCSC3)=O)CC2)=O)cncc2ccccc12 C(C)(C(=O)N(C1CN(C(=O)CC2(CN(C)C)CCC2)C1)C)OC C1(NC(c2c(C)nc(CC(C)C)s2)=O)CCCCN(Cc2cscn2)C1 CC1C(=O)CCC1CC(N1CCC(OCC(=O)NCc2cccc(Cl)c2)C1)=O c1(OC)cccc(CC(=O)NCC(C)CNC(=O)C(C)NC(C)=O)n1 C1(COC)(CNC(=O)CC2CC2)CCN(C(C2(Cl)CC2)=O)C1 C12(C(=O)NC(C)(C)CC(F)(F)F)C3CC(CC13)C2(F)F N1(C(C2CCC(C)C2)=O)CC2N(C(=O)CC3CC4(CCC4)C3)CCC2(C)C1 CCC(CNC(=O)Cn1nccc1C)(CC)C(=O)NC1(CF)CCC1 c1(C(N(C)C)=O)cncc(C(=O)NC2CC(N(C(=O)CN(C)C3CC3)C)C2)c1 CP(C)(=O)C(O)C(=O)N1CCC(O)(CNC(c2cnoc2C2CCC2)=O)CC1 C(C(C)(O)CNC(=O)Cn1nnc(-c2cccs2)n1)NC(CC1(CSC)CC1)=O c1(CC(C)NCc2ccc(N3CCOC(C)C3)nc2)cccc(O)c1 Cc1c(C(=O)NCC2CCCN(C(c3cc(CCO)on3)=O)C2)cncc1N N1(C(c2cc(C)no2)=O)CCCC12CCN(Cc1cnc(Cl)nc1)CC2 N1(C(C(CC2CC2)NC(C=C(CCC)CCC)=O)=O)CCCOC(C)C1 C=C(Cl)C(C)(C)C(=O)NCC(C)CN(C(=O)Cc1cncn1C1CC1)C c1(C(=O)OCc2scc(C)n2)ccc(F)c(Cl)c1.N12CCCC1C2=O C(CC(C)C)(C(=O)NC1CCCCC1C(N1CCCC1C(=O)N(C)C)=O)OC C1(C(=O)NCCC2CC(F)(F)CN2C(c2cc[nH]n2)=O)CS(=O)(=O)CC12CCC2 c1(N2CCCC(NC(=O)C(F)(F)c3ccccc3)C2)ncnc2[nH]ccc12 CCCN=C(NCC1CCCN1C(=O)OC(C)(C)C)NCC1C=CC2CC1CO2 c1(N(CCN2CC(C)OC(C)C2)CC2CC2)cc(S(C)(=O)=O)ncn1 C1(C(=O)NC2CCC(OC)C2)CC2CC1CN(C(c1csc(=N)[nH]1)=O)C2 C#CC1CC2(CC2)CN1C(=O)CCC1CCCN(C(c2cc3n(n2)CCC3)=O)C1 c1(CC)cc(C(N2CCC(C)C(NC(c3ccc(NC)nn3)=O)C2)=O)ccc1F c1(CC(=O)N(C2CCN(C(=O)CCC(C)N(C)C)CC2)CCC)ccnnc1O S(=O)(=O)(c1ccc(SC(F)(F)F)cc1)NC(C(C)C)COC(C)(C)C C1(C2CC2)(C(=O)NCc2cn(C3CCN(C(C=CCN(C)C)=O)C3)nn2)CCC1 N1(C(CNC(N)=O)=O)CCN(C(=O)Nc2cc(F)cc(F)c2)CC1CCO C1(CNC(CN(C)C(C2CCCCO2)=O)=O)C=CCN1C(=O)COCP(C)(C)=O C1(C)(C(=O)NC(CN(C(=O)Cc2cn[nH]c2)CC)C)CCCN(C(C)=O)C1 C(=O)(CC(C)C(C)C)N1CC(OC)C(C(=O)Nc2ccc(SC)nc2)C1 c1(CC(=O)N(C2CCc3c[nH]nc3C2)C)ccc2c(c1)CCCS2 C1(NC(=O)COC2CC(F)(F)C2)CN(C(C2CN3CCC2CC3)=O)CC2CC12 C1(CCC(=O)NC(CNC(CCN(CCCCOC)C)=O)CO)CCCCCC1 c1(C(N2CC(NC(c3nc(OC)oc3)=O)(CO)C2)=O)cccnc1C(F)(F)F C1(CNC(Cc2c(C)noc2Cl)=O)CC2CCCC2N1C(=O)C(F)C1CCCC1 C(CC(O)C(=O)N(C)CC1CCC(=O)N1)NC(COC1(C#C)COC1)=O c1(C(N(C)CCNC(c2cccc3ncnn23)=O)=O)nc[nH]c2ncc(Br)c1-2 c1(C(=O)NC2C(NC(c3ccnc(CO)c3)=O)CCC2)cnc2sccn12 N1(C(C(CC2CC2)OC)=O)CC(C(=O)N(C)C(c2ncccn2)C)CC(C)(C)C1 C1(NC(c2occ(C)c2)=O)C2CC1CN(C(=O)CCOc1ccccc1F)C2 N1(C(C2(C#N)CC3CC3C2)=O)CC2CCCC2(C(=O)Nc2ccc(Cl)cc2O)C1 C1(NC(=O)Nc2cc(C)nc(C)c2)C2CCOC2C12CCCC2 C(=O)(N=c1[nH][nH]c(C)c1Cl)C1C(NC(c2c(C)nc[nH]2)=O)CCC1 C(CCC(=O)NCC1COC(CNC(=O)CSc2nncn2C(C)C)C1)SC N1(C(CCC)=O)CC(F)(F)CC1CNC(c1cc(C2CC2)on1)=O Cc1ccc(C(=O)NCC2(O)CCN(C(C3CCC(C)S3)=O)CC2)c(C)c1 C1(Cn2cc(C(CC(=O)OC)(C)C)nn2)CCN(C(=O)C(C)(C)O)CC1C c1(-n2cc(C3C(NC(C(c4n(CCC)ccn4)(F)F)=O)C3)nn2)ccc(Cl)cc1 CCC(CCC(=O)NCc1ccc(C)c(C)c1)NC(c1cc(C#N)n(C)n1)=O C1(C)(C(=O)NC(C)CC2CN(C(c3c[nH]ccc3=O)=O)CCO2)CCN(C)CC1 CCC(C)(C)C(=O)N(C1CC(NC(C2COCCN2CC2CCC2)=O)C1)C c1(C(=O)NC2C(NC(c3nc(C)oc3)=O)CC(F)(F)C2)c[nH]c2nc(Cl)ccc12 C1(CNC(CCCCOCC)=O)CN(C(c2c[nH]cc2C2CC2)=O)CC(C)(C)O1 c1(CN(C2CN(S(=O)(=O)c3ccc(Br)s3)C2)C)ccnc2c1ccc1cccnc21 N1(C(C2(C#C)CCC2)=O)CCC2(CCN(C(c3c(F)c(C)cc(N)c3F)=O)C2)C1 C1(C(=O)NC2CCN(C(C3CC4=C(C3)OCCO4)=O)C2)CC2C=CC1CCC2 c1(C(=O)OC)ccc(NC(C2(C)CCCN2C(=O)CSC)=O)c(F)c1 C1(CNC(C2(c3ccccc3)CC2)=O)CCCN1C1CC1 C1(NC(CSC)=O)CCCCCC1NC(=O)CCc1nc(C)no1 N1(C(C(F)OC)=O)CC2(CCOCC2)CC1CNC(=O)C=CC(N)=O N1(C(C2(C=C)CCN(C(c3ncccc3CC)=O)C2)=O)CCC(C#CC)CC1 C1(C(C)NC(=O)COc2cn[nH]c2)CCN(C(c2cnc[nH]2)=O)C1 C1(C)(NC(CNS(NC)(=O)=O)=O)CCN(C(c2ccc(Br)c(Cl)c2)=O)CC1 c1(C(=O)NC(CCCNC(CN(C(C(C)C)=O)C)=O)C)cccc(F)c1C1CC1 c1(OC)cc(C(=O)NC2CCC2C(=O)NCC#CC2CC2)nn1C n1(CC)nnc2cc(C(=O)NCC3COCCN3C(C3CC=CCO3)=O)ccc12 C1(N(C(CCCCCC)=O)CCC)CC(O)C12CCCC2.C(C)(C)(C)O C12(CC(N3CCOCC3C(F)F)=O)CCC1CN(C(C1CCC(C3CC3)C1)=O)C2 CC1CCCCC1(CNC(=O)COc1cccc(C#N)c1)NC(=O)CCCF C(c1cccc(Cl)c1)=C(C)C(=O)NC(C)(CNC(=O)C(F)C(C)C)C(C)C C(=O)(C(C)(O)c1ccccn1)N(CCN(C)C(c1cccnc1)=O)C c1(C(=O)NCC2COCCN2C(C2CC(CF)C2)=O)cccc2[nH]ncc12 C1(S(C)(=O)=O)(C(=O)NCC2CCN(C(C(Cc3c(C)nc[nH]3)O)=O)C2)CC1 c1(C(=O)NC2CCC(NC(CCCOC(C)C)=O)CC2)c(F)cc(Cl)cc1F C1(C)(CNC(CC2(C)CCN(C(C(CC)COC)=O)C2)=O)CCC(=O)N1C N1(C(C(COC)C)=O)CCC(C2(NC(C3CC(C)(C)OC3(C)C)=O)CCC2)CC1 c1(CN2C(C(N3CC(C(=O)OC)C3)=O)CC3CC32)cc(Cl)ccc1Cl CC1(C)COCCC1C(=O)NCC1CC2CCC1N2C(=O)C(C1CCOCC1)O C(=O)(C(CO)C(C)(C)C)N1C(CNC(C2CCC(C)(C)CC2)=O)CC(F)C1 C1(CNC(=O)NCC2(F)CCC(F)(F)C2)(CO)COCC2CCCN12 C(=O)(C#CC1CCOCC1)N1CCC(CCNC(CC(C)SC)=O)C1 C(=O)(C(F)(F)C(O)CC)N(CC(CC)NC(c1cnn(CCO)c1C)=O)C N1(Cc2cc(OC)ncc2)CCC(NC(=O)CCc2cccs2)CC(C)(C)C1 CCCC(CC(=O)NCCCOC1CCC1)NC(=O)C(F)(F)C(C)O c1(C(=O)NCC2CN(C(COC(CC)C)=O)C(C)(C)C2)ccc(O)cc1[N+](=O)[O-] C(C)(C)(CC(=O)NCC1(C)CCCCC1)NC(C1C(C)(C(C)C)C1)=O N1(C(c2c(CC)onc2)=O)CCC(CN(C(c2sncc2C)=O)CC)CC1 N1(C(C(CCOC)C)=O)CCC(C)(NC(c2ccsc2C)=O)CC1 C1(C(=O)NCC(C)(CO)NC(=O)C=Cc2cc[nH]n2)CCn2nnnc2C1 C=CCC(CNC(C1CCCC(=O)N1)=O)C(=O)N(CC(C)(F)F)C N1(C(C(CCC)OCC)=O)CCC2(CCN(C(c3cnn(CC)c3C)=O)CC2)C1 c1(C(=O)NCC(C)(C2CCC2)NC(COc2cn(C)nc2)=O)[nH]cc2c1CCC2 n1(C(C(N2C(CNC(CN(C3CC3)CC)=O)C=CC2)=O)C)cnc2ccccc12 N1(C(C2(C(C)C)CCOCC2)=O)CCN(C(c2cc(N)ccc2Cl)=O)C2(CC2)C1 C1(CNC(=O)COC(F)(F)F)CC2(CN1C(=O)CC1CC=CCC1)CC2(F)F C1(C(N2CCC(C)(CNC(c3ccnn3C(F)F)=O)C2)=O)CCC2(CCC2)O1 Cc1ccc(Cl)c(C(=O)NC2CC2NC(c2cn(C)ccc2=O)=O)c1 CCCCS(=O)(=O)CC(=O)NC1CCC(CCNC(C2CC23CC3)=O)C1 C(=O)(C(C(C)(C)C)N(C)C)N1CCC(O)(C(C)NC(=O)CC2CC(F)(F)C2)C1 c1(CC(=O)N(CC(C)NC(=O)COC2CCN(C)CC2)C2CC2)ccc(F)nc1 C1(C)(CNC(C(C)(C)N(C)C)=O)CCN(C(=O)CCC(=O)Nc2nccs2)CC1 N1(C(CC(CC2CC2)NC(c2c(CC)noc2C)=O)=O)CC2C(C1)C2(F)F c1(CNC(CC2ON=C(CC)C2)=O)ccc2c(c1)CN(C(c1cscc1C)=O)C2 N1(C(C2CC(C)C2)=O)CCC(C)N(C(c2n[nH]c3ccccc23)=O)CC1 c1(C(=O)NCC2CN(C(C(C)c3ccco3)=O)CC2O)ccc2c[nH]nc2c1 CCC(C)CC(C)CC(C)C(=O)NNC(=O)Cc1csc(N2CCOCC2)n1 CC1CN2CCN1CC2C(N1CCC(OCCCNC(=O)C2=CCOC2)CC1)=O c1(C(N2CCCC(NC(C34OCC(C(C)C)(C3)C4)=O)C2)=O)c(Cl)ccc(F)c1N C1(C(=O)NC(C(=O)OC)Cc2csc(Cl)c2)C2Cc3cc(Br)ccc3C12 C(c1ccc(C)nc1)=CC(=O)N(C1(CC=C)CCN(C(=O)C(CC)CC)C1)CC Cc1nc2ccccn2c1C(=O)Nc1noc(-c2cc(Br)cnc2O)n1 c12cnccc1NC2=O.c1(CN(C(C=CC)=O)CC)cccs1 C(=O)(C(O)C(C)(C)CC)NCc1cn(CC(=O)NC2C(C=C)COC2)nn1 Cc1ccc2c(N(C)Cc3cccnc3)nc(N(CC(=O)N(C)C)C)nc2c1 C1(C2(O)CCC2)(C(N2CCCC(CN(C(C3N(CC)CCOC3)=O)C)C2)=O)CC1 CCC(C)(COC)C(=O)NC1COCCN(C(=O)Cc2ccccc2OC)C1 C1(NC(CCOCC)=O)CN(C(C2(F)CCC(C)CC2)=O)CC1(C)C c1(OC)ccc(Br)c2cc(C(=O)NC(C(=O)O)C(F)(F)F)[nH]c12 Cc1cc(C(=O)NC(C)CC(C)NC(=O)C=Cc2cccnc2C)c(N)c(F)c1 N1(C(C(OC)OC)=O)CCN(C)C(C(=O)NCCc2nnc(O)o2)C1 N1(C(Cn2ncc(CC)c2)=O)CCc2sc(-c3cnc(C)s3)nc2C1 C1(OC)CN(C(c2c[nH]c(Br)c2)=O)CC1NC(=O)C(C)SC N1(C(CCC2C(C)(C)C2)=O)CC2CCCN(C(=O)C(O)C3CCCC3)C2C1 C1(NC(c2cc(C)sn2)=O)CCSC12CN(C(=O)CCCC(F)(F)F)C2 C1(CCC)CCCCN1C(=O)NC(c1csc(-c2ccc(Br)cc2)n1)C C1(C(N(CCC(=O)OC)CC)=O)CSCN1C(=O)Cc1ccoc1C S(=O)(=O)(c1ccccc1F)N1CCC(NC(Cc2c(OC)cc(Cl)cc2)=O)CC1 C=CC(C)(CC)C(=O)NC1CCC(CNC(=O)C(C)C(=O)OC(C)(C)C)CC1 C1(COC)(NC(=O)Cc2nccn2C)CCN(C(c2cccc(C(N)=O)n2)=O)C1 N1(C(C2(CCC)CCC2)=O)C(C(=O)NCC(c2ccnn2C)O)CCC12CC2 CC(CC(F)(F)F)NC(=O)CC1(C=C)CN(C(c2cnncc2O)=O)C1 C(=O)(CCCS(C)(=O)=O)NCC(C)(C1CCC1)NC(Cc1nnc(C)o1)=O CCC(C)CC(C)C(=O)NC1(C(=O)NCC(F)(F)C(C)(C)O)CC1 C1(NC(c2coc(Br)c2)=O)CCN(C(C2CC(F)(F)C2)=O)CCC1(F)F C1(NCCCCC)CCC(C(=O)NC2CCN(C(=O)CSc3nncn3C)C2)C1 N1(C(C2CC(C)=C(C)CC2)=O)CCC2C(C1)CN2C(c1ccc(O)nc1)=O O=C1CCc2cc(NC(C3(O)CN(Cc4cc(Cl)ccc4Cl)C3)=O)ccc2N1 C1(Cn2c(CC)nnc2N(C)CCc2ccc(Cl)c(F)c2)CC2C(C1)C2(F)F c1(CC(N2C(C(N(C3(C#C)CC3)C)=O)C(CC)CC2)=O)ccccc1C#C N1(C(COCc2cc(C)on2)=O)CCN(C(=O)CCCCN(C)C)C2COCC12 C1(NC(C(C2CCCC2)OCC)=O)CC(C)(NC(=O)Cc2ccc(Cl)s2)C1 C(=O)(C(F)(F)CO)NC(C)C(C)NC(c1n[nH]cc1F)=O N1(C(C2(OCC)CCC2)=O)CC2CCCC(NC(=O)C(C3CCOCC3)C)C2C1 C123COCC1CN(C2)N1CCCC(CC1)C3C.C(=O)CCn1cccc1 Cc1cc(=N)[nH]cc1C(=O)NC1CC(NC(c2cnc(O)c(Cl)c2)=O)C1 c1(OC(C)C)ccc(C(N2CCCC(CCNC(=O)C(C)(F)F)CC2)=O)c(Cl)c1 C1(C(N(C2CCN(C(COC)=O)C2)CC2CCSC2)=O)CN(C)CC(C)O1 Cc1cc(N2CCC(N3CCSC(=O)CC3)C2=O)cc(Br)c1 C1(C(=O)NCC2N(C(CCc3ccc(OC)cc3)=O)CC2)CC(=O)NC(=O)C1 C1(CNC(C2C3COCC23)=O)CC2COCC2N1C(c1cccnn1)=O c1(CC(=O)NCC2CC(C)N(C(=O)Cc3cnc[nH]3)C2)cnc2ccccn12 c1(C(=O)NC(C(C(=O)N(CC(=O)N(C)C)CC)C)C)cccc(O)c1C N1(C(C2(C3(O)CCC3)CCC2)=O)CCCC2CCC12CO CC1OCCCC1C(=O)NCC1C2CN(C(=O)CCc3cnn[nH]3)CC12 C(=O)(C(CC(C)C)NC(=O)CC1CCCC2CC12)NCC(C(CC)C)C C12(C(N(CCCSC)C)=O)COC(CC3CC3)(C1)C2.C12(CC1)CC(=O)N2 C1(C(=O)NC2CCN(Cc3ccc(-c4nn[nH]n4)cc3)CC2)CC2(CNC2)CO1 CCC(CC)C(F)C(=O)NCC(C(=O)NC1CCCNC1=O)C(C)(C)C c1(C(=O)NC2(CC(=O)N(CCNC=O)CC)CC2)c[nH]c(=NC)s1.CC1CC1 C(=O)(C(C)C(C)CC)NC(CCNC(c1ccc(CCC)[nH]1)=O)C Cn1c(C#N)cc2c1CCN(S(=O)(=O)CCCC(C)(F)F)C2 N1(C(C=C2C(C)(C)CCCC2)=O)CCCC12CCN(C(=O)CS(C)(=O)=O)C2 C(=O)(C(O)C(C)(C)C)NCCC1(C(=O)NC(c2nn[nH]n2)CC)CCCC1 C(=O)(CC(C)(F)F)N(C(CCNC(C1(CCOCC)CCCC1)=O)C)C N1(C(C2(CC#C)CCCCO2)=O)CC2(C1)CN(C(=O)Cc1ccnn1C)C2 c1(OC)cc(CC(=O)NCc2ncc(C(=O)O)[nH]2)ccc1F N1(C(c2c(C)[nH]nc2Br)=O)CCCN(C(=O)CCC2CCCN2C)CCC1 CON=CC(=O)NCC1CCCN1C(c1csnc1OC)=O CCC(C)C(O)C(C)C(=O)NCCCC(C)(C)NC(=O)CCc1csnn1 Cc1cccc(F)c1C(=O)N(C(C)C(=O)NC(C)(CO)CC(C)C)C1CC1 C1(C(COC)C)CCN(C(=O)NC2CC(F)C(=O)N2)CC1 CCCCC(O)C(=O)NCc1cc[nH]c1C(=O)NC(CO)C(C)(C)C C(c1nc2ccccc2[nH]1)=CC(N1CC(CNC(C(C(C)C)F)=O)C1)=O C(C(C)(C)CC(=O)N1CCOC(C(N)=O)C1)NC(c1ccc(C#C)o1)=O C1(N(CC(N2CCC(n3cc(C(CC(C)C)O)nn3)C2)=O)C)CCCC1C#N C1(NC(c2c(C)n(C3CC3)cc2)=O)CN(C(=O)CS(C)(=O)=O)CC12CC2 CCCCC(C)(CO)NC(C1CCN(C(c2nonc2C)=O)C1)=O C(=O)(C(F)(F)CN1CCCC1)N(CC(CNC(C1(OC)CCCC1)=O)(C)C)C CC1CCC=C1C(=O)N1CCN(C(=O)CCF)CC1CO C#CC1CCCCN1C(=O)CCC(CC)NC(=O)CNc1cccnc1 c1(CCCC2N(Cc3nc(CC(=O)NCCC)on3)CCC2)cccnc1Br c1(C(=O)OCC(c2cn(CCC)nc2)=O)c[nH]c(C)c(Cl)c1=O C(=O)(C1=NOC2COCC12)N1CCC(C)(CC(=O)NCC(=C)CC)C1 c1(C(=O)NCCNC(C2C(C)(CC)C2)=O)ccc(S(=O)(=O)C2CCC2)cc1 C1(CNC(C2(CNC(c3ccc(OC)cc3)=O)CC(=C)C2)=O)C2CCCCC12 Cc1cc(C(=O)NCC(C)(O)CNC(C2CS(=O)(=O)C2)=O)cc(C)c1C#N c1(CC)cc(C(=O)NCC2(CNC(=O)C(C)(C)c3csc(C)c3)CC2)c(C)o1 CCCC(C(O)C(=O)NCC(C)(C)O)NC(C1(CC2CC2)CC1)=O c1(C(N(CC(CNC(C23CC(CC)(C2)C3)=O)O)C)=O)sc(N(C)C)nc1Cl c1(C(N2CCCC(NC(C3CCOC3)=O)CCC2)=O)cccc2sc(O)nc12 Cc1ccc(F)c(C(=O)NC2CCCN(C(=O)CC3CCC(=O)O3)CC2)c1Cl c1(C(=O)NC(C)C(CO)NC(=O)C2=CCCS2)ccc2nc(N(C)C)[nH]c2c1 C1(OCC)CC2(C1)CC2Nc1cc(NCCC2CCN(C)C2)ncn1 c1(C(=O)OCc2cc(C)c(Br)nc2)nc(C2CC2)n2ccccc12 c1(NCCCCC(C)NC(CCn2c(C)csc2=O)=O)ncc(Cl)cc1[N+](=O)[O-] C(=O)(CC(C)(C)O)N(CCCNC(C1(CC)COC1)=O)CCO C1(C(=O)NC2(CF)CCN(C(c3c(C)cc(C)[nH]3)=O)C2)CCc2nn(C)cc2C1 CCC(C)C(O)C(=O)NCC1COCCN(C(c2sc(COC)nc2C)=O)C1 Cc1ccc(NC(c2coc(C3CC3)n2)CSc2ccccn2)cc1 Cc1cccc(Br)c1C(c1nnnn1C1CC1)NCC1CC(O)C12CCC2 N1(C(c2c(C)oc(C(C)C)n2)=O)CC2(CC(NC(=O)COc3ccsn3)C2)C1 N1(C(C(CSC)C)=O)CCC(CNC(C2(c3ccc(F)cn3)CC2)=O)C12CC2 C1(C(=O)NCC(C)N(C(=O)C=Cc2nnn(C)n2)C)CCCCN1C CC1CCC(NC(C2(C)CCC2)=O)CN1C(=O)CO C1(NC(=O)NC(C(=O)NC(C2CCCC2)C)Cc2ccoc2)CCCC(CO)C1 Cc1nnc2n1C(C(=O)NC1CC(CNC(C3CCCN3C3CC3)=O)C1)CC2 C1(C(=O)NC(CN(C(c2cc(Br)c(C)o2)=O)CC)C)(COC)CC=CCC1 N1(C(Cc2ccc(C(C)=O)s2)=O)CCN(C(C2CCCC(O)C2)=O)C2(CCC2)C1 c1(C(=O)NCCCCNC(=O)COCc2ccccc2)ccc(N2CCC2)nc1 C1(NC(C2(SC)CC2)=O)CC2CCC1N2C(=O)C1=NOC(c2ccc(F)cc2)C1 C12(NC(=O)C3=CCCC3)CCN(C(C34CCN(CC3)CC4)=O)CC1C2 c1(C(=O)NC(CC(C)NC(c2cc(SC)c(C)o2)=O)C)cn2c(n1)CCC2 N1(C(C(CN(C)C)(F)F)=O)CCN(C)C(CNC(=O)CCCc2nccs2)C1 N1(C(c2c(CCC)n(C)nn2)=O)CCC(C)C(NC(=O)CCc2ncccn2)C1 c1(C(N(C)CC2CCCN(c3nccc(C#N)n3)C2)=O)ccc2ccn(C)c2c1 C1(C(N2CCC(N(C(C3C(C(=O)OC)CCCC3)=O)C)C2)=O)CC(F)(F)C1(C)C c1(OCC)ccc(Cl)nc1C(=O)NCC1(F)CC(NC(C2CCC(F)C2)=O)C1 C=CCCCC(C(=O)N1CCC(CC(=O)OC)C1)C1C2CCCC12 N1(C(CCc2c(C)ncs2)=O)CC(CNC(c2csc(CO)n2)=O)CC1(C)C C1(OC(c2c(N)cc(O)cc2F)=O)CCc2ccccc2C1=O c1(C(N(C2CC(NC(=O)C=CSc3ccccc3)C2)C)=O)ccsc1S(N)(=O)=O c1(C(=O)NC2CCC(N(C(c3c(OC)csc3)=O)C)C2)cc2ccccn2c1 C1(NC(CC(CC)C2CCC2)=O)CC=C(C(=O)NCCC2CCOC2)C1 c1(OC)ccc2c(n1)NC(C(N1CCC(CCNC(=O)CC(C)O)CC1)=O)C2 c1(C(=O)OC(=O)NC2C(CC)C2)ccc(SC)cc1.c12ccc(cc1)[nH]c2=O C1(CNC(CNC(=O)NC)=O)CC(NC(c2nccc(N)c2Cl)=O)C12CCC2 N1(C(CCC2C(C)(C)C2)=O)CCOC2(C1)CN(C(C1(c3cccs3)CC1)=O)C2 c1(C(=O)NCc2cccc(CNC(C3C(C)(CC)C3)=O)c2)ccc2nnnn2c1 c1(C(N2CCC(F)(CNC(=O)COCC3CC3)C2)=O)ccc(F)c(CO)c1 C1(NC(c2cnc(COC)s2)=O)CN(C(C2C3COCC23)=O)CCC1CO C1(NC(C(C)C2CC2)=O)CCC2(CC1)CN(C(c1cccc3[nH]nc(O)c13)=O)C2 c1(OC)ccc2cc(C(=O)NCC(C)N(C)C(c3cc(CF)on3)=O)ncc2c1 c1(C(N(CC(C)NC(C(CC)OC)=O)C)=O)cncc(N)c1 Cc1nc(CCC(=O)NC2C=CC(CNC(=O)C(F)n3cccn3)C2)cs1 Cc1nc(C(=O)NCC2CC(NC(c3ccnc(C(F)(F)F)n3)=O)C2)c(C)n1C c1(C(N(CCN(C)Cc2cn(Cc3ccc(Cl)s3)nn2)C)=O)nc(Cl)c(Cl)s1 Cc1c(C(N2CCC(NC(=O)C(F)C3CCC3)C2C)=O)[nH]c2c(Cl)cccc12 c1(C(=O)NCCC2CC(NC(C3(C)COC3)=O)C2)cc2ccccc2oc1=O N1(C(C(COC)O)=O)CCC(CO)(CNC(=O)C=Cc2ccc(C)o2)C1 c1(N2CC(CC(C)NC(c3c(CC)n[nH]c3)=O)C2)ncc2c(n1)CCOC2 C1(NC(=O)CCC2CCCO2)CN(C(=O)C2=COCC2)CC(F)(F)C1 c1(C(=O)NCC2(F)CC(NC(c3ccc(C)n3C)=O)C2)csc2ncnc(O)c12 c1(CNCC2OCCN(S(CCCC)(=O)=O)C2)cc(F)ccc1OC N1(CC(=O)NCCC2CC(NC(C(C)=C(C)C)=O)C2)CC2CC2C1 CCC1=NOC(C(=O)NCC2COCCN2C(c2nc(C(F)(F)F)sc2C)=O)C1 CCCC(C(=O)N1CC(N(C)C)C(C)C1)NC(=O)C=CC(=O)N(C)C CC1(C(N2CC(CNC(C3(n4nccn4)CC3)=O)C2)=O)C2Cc3ccccc3C12 CC(C)CC(C)(CNC(c1ncccc1Br)=O)NC(C1CCC(O)C1)=O c1(OC)c(C(=O)NCC2CCN(C(c3cnc(O)c(F)c3)=O)CC2)cccc1F Cc1cnc(C)c(C(=O)NCC(C)(O)CNC(C2CC(F)(CO)C2)=O)c1 N1(C(c2ccc(CC)cc2)=O)CCC(C)C(N(C(=O)Cn2ccnn2)C)C1 C1(NC(CCC(=O)N(C)C)=O)CC12CCC(NC(C1CCCC1(F)F)=O)CC2 CCCCCCC(=O)NC1CCCN(C(c2ccc(F)s2)=O)CC1 C(=O)(CP(C)(C)=O)N(C1CCC(NC(C2(OC)CCCC2)=O)C1)C CCC(CC)C(C(=O)N1CCC(CN(C)C(C2CCCCC2)=O)C1)OC c1(OC)cc(NC(C2CSCN2C)=O)c(Cl)c(I)c1 C1(C(=O)NCC(C)Sc2ccccc2)CC(=O)N(Cc2ccc(Br)cc2)C1=O C1(=CCNC(c2c(CC)c[nH]c2)=O)CCN(C(C2OC(C)CC2C)=O)CC1 Cc1cn(C)nc1CC(=O)NCC1(NC(=O)COC(C)C)CCOC1 C1(OCC)CN(c2ccccc2)CC1CNC(=O)COCC.C1(C)(C=O)CC(C)C1 C(C(C(=O)N1CCC(CF)C1)NC(=O)COC1CC(F)(F)C1)OCC Cc1c(CC(=O)NCC(C)NC(=O)CC2(N(C)C)CCCC2)cccc1Br Cc1ccsc1C=CC(=O)NC1CC(N(C(=O)C=CCCc2ccccc2)C)C1 c1(CNC(C(CCC)=CCC)=O)ccc2c(c1)CCN(C(=O)CC(C)C(C)C)C2 CN1C(=O)CCC1CC(=O)NCC(N1CCN(C(=O)CC2CN(C(C)=O)C2)CC1)=O N1(C(C(C(C)OC)N(C)C)=O)CCC(CO)C(NC(=O)CC2CCCC(C)O2)C1 c1(OCc2ccco2)ccc2cccnc2n1.C1(OC)CC2N(C1)CCN(CC)C2 CC1CN(C(c2cccc(C(N)=O)c2)=O)CCC1CNC(=O)Cn1nnc(=N)[nH]1 c1(OCC)cccc(C(=O)NC2(CNC(C3CCCO3)=O)CCCCCC2)c1N C1(F)(C(N2CCC(OCC)C2)=O)CCN(c2ccncn2)C1.C(C)(C)C C(=O)(C(F)C(F)(F)C(F)(F)F)NCCCCCCNC(C=C(CC)CC)=O N1(C(C2CCOCC2)CC)CCCC2(CCN(C(C3(C(=O)OC)CCC3)=O)C2)C1 C1(NC(=O)CC2CCCC2)CCC12CCN(C(C1CS(=O)(=O)C1)=O)CC2 C(=O)(CC(C)CC(C)(C)C)NCCC(C)NC(c1ccc(COC)o1)=O c1(C(=O)NC2CN(C(c3cc(OCC)n[nH]3)=O)CC2O)cc(C)ccc1F c1(C(=O)NCC2CN(C(C3CCCCO3)=O)CCO2)ccc(O)c(F)c1 Cc1c(F)ccc(C(N2CC3CC3(NC(=O)C(C)CC3CC3)C2)=O)c1C C=CCN=C(NCc1cn(CC)nn1)NC(c1ccco1)C C#Cc1cccc(C(=O)NC2CCCN(C(=O)CC3(N(C)C)COC3)C2C)c1F CCC(CC(=O)N1CCCC1C1(NC(C2CN(C(C)=O)C2)=O)CC1)CC(F)(F)F c1(CCCNC(CN(C(=O)CCCC2CCC2)CCOC)=O)nncn1C c1(C(N2C(C)C(NC(C3(c4cccnc4)CC3)=O)CC2)=O)cc2ccsc2n1C C1(C)(COC)CC(NC(=O)CNC(C)=O)CN1C(c1cc2n(c1)CCC2)=O c1(OCC)ccc(CC(=O)N(C2CCN(C(C3(C)CCCOC3)=O)CC2)C)cc1 c1(C(C(N2C3C(NC(C(C)CO)=O)C(C3)C2)=O)=O)cc(S(N)(=O)=O)cn1C N1(CC)OCC(OC(=O)C(c2ccccc2F)F)C1=O Cc1ccnn1CC(=O)OC(C)C(=O)NC(C)(C)C C(=O)(CCCCCCN=[N+]=[N-])N1CCCC(F)(CNC(C(CC)O)=O)C1 N1(C(C2C(C=C)OCC2)=O)CC=C(CNC(=O)C(C)(F)F)CC1 c1(CCC)[nH]nc(C(=O)NC2CCN(C(=O)Cc3ccc(C)nc3)C2)c1[N+](=O)[O-] c1(C(N2CC(CCCC)N(C(=O)C(C)CSC)CC2)=O)cc2ccccc2o1 CC(c1ccccc1C)=CC(=O)NCCC(C)NC(c1coc(CC2CC2)n1)=O C(=O)(C1=CS(=O)CCC1)NC(C1CCCC1)CNC(C(C(C)C)N(C)C)=O n1(CC(C)C)ccc(C(=O)N(CC(O)CNC(=O)CC2CC(CF)C2)C)cc1=O C1(C(N2CCN(C(c3cccc(C)c3N)=O)CC2CO)=O)CC2CCC(C1)C2O C1(COCC(=O)NC2CC2)(CO)CCN(C(=O)CC2(C(c3ccncc3)C)CC2)C1 C(=O)(C1CCCn2nccc21)N1CCCN(CCNC(C(=O)NC(C)C)=O)CC1 CC(CC(=O)Nc1cccc(C(=O)NC2CCC([N+](=O)[O-])CC2)c1)C(C)(C)C c1(C(N2CC(C(=O)NCCCC3C(C)C3)CC2(C)C)=O)c[nH]c2ncccc12 C1(C(C(=O)NCC2CC2NC(=O)Cc2ccco2)OC)CC(F)(F)C1 C1(C(=O)Nc2cc(OC)c(F)cn2)CCCC12CCN(Cc1cc(Br)co1)C2 N1(C(C=CCOC)=O)CC2(CCN(C(=O)CN3CCNC(=O)C3)CC2)CC1C CC1(C)OC2CC(C(=O)NC3(CO)CCN(C(=O)CCN4CCC4)C3)CC2O1 c1(C(N2CCC(C)(CNC(C3(Cl)CC34CCC4)=O)C2)=O)cc(N)c(F)cc1F C#CCCCCCCCC(=O)NCCN(C)C(C1CCNC1=O)=O C(=O)(CCS(C)(=O)=O)N(C)CC1(NC(C2CC(=C(F)F)C2)=O)CC1 c1(C(=O)NC(CC)CNC(c2cnc(N(C)C)nc2)=O)cc2cccnn2c1 C1(NC(C2CC(SC)C2)=O)CC2CC(NC(=O)CC(C)C(C)C)C1C2 C12(C(=O)NCCSCC=C)CC(CN(C(=O)CCCC(=O)C3CC3)C1)C2 C1(C(=O)NC2CC(C(N(CC(COC)(C)C)C)=O)C2)C2CCC(F)(F)C12 Cc1c(C(N2CCCC2CNC(c2cn(C)nc2C2CCCO2)=O)=O)ccn1C c1(C(c2n(CCC(=O)OCC)nnn2)Nc2cn[nH]c2)cc(OC)c(O)cc1Br N1(C(C2CCCC(OC)C2)=O)CCCC(NC(c2cnn(CCO)c2)=O)C1C c1(C(=O)NCC(CCNC(c2n(CC=C)ccc2)=O)O)cc(N(C)C)ccn1 c1(OC)nc(=NC2CCCC(C(=O)Nc3cc(C)c(F)cc3C)C2)[nH]cc1C#N N1(C(Cc2ccn(CC)n2)=O)CC(NC(=O)CC23CCCC2C3)C2(CCCC2)C1 N1(C(C=COCC)=O)CCN(CCOC2CCN(C(=O)C(C)C)C2)CC1 C(N=c1cc(C2CC2)nc[nH]1)C1N(C(c2cc(SCC)ncc2)=O)CCCC1 CC1(C)CC2(CC(C(=O)NCC3COC(CNC(C4(Cl)CC4)=O)C3)C2)C1 c1(-c2cc(C)c(C#N)cc2)ccc2ncc(C(=O)Nc3ncc(C(C)C)s3)n2c1 N12CCCC(CC1)N(C)C2=O.c1(C(C)C)noc(CSc2nc(C3CC3)no2)n1 C1(NC(c2nc(C)sc2)=O)CC12CCN(C(c1ccc(N)cc1Cl)=O)C2 N#Cc1cc(C(=O)NC2CC(CNC(C34CCCC3C4(F)F)=O)C2)c(N)nc1O c1(CC(=O)NC(C)C(C)NC(C2(N3CCCC3)CCC2)=O)nnc(S)s1 Cc1cccc(CC(=O)NCCC2CCN(C(C3CCC4CC4CC3)=O)C2)c1C C(=O)(C1=CCCSC1)NCCN(C(c1cnc(C(C)=O)s1)=O)C N1(C(COC2CC(NC(C3CCCC34CCC4)=O)C2)=O)CC2CCCC(C2)C1 C1(C(NOCCN(C)C)=O)CCCC1CNC(C1CCCC1F)=O N1(C(CSSC)=O)CCCC(NC(c2c(C)nsc2N)=O)C1C CC1CCCC1C(=O)NCC1(O)CC(CNC(=O)CC2CCCC2)C1 C1(C(N(CC(C)CNC(c2cscc2Br)=O)C)=O)Cc2nncn2C1 c1(C(=O)NCc2ccc(CN(C(C(CC)F)=O)C)cc2)cnc2n1CCCC2 C1(C(=O)NC(C2(O)CCN(C(c3ccc[nH]3)=O)CC2)C)Cc2nccn2C1 c1(OCCC)ccc(C(=O)N(C)CCOCCN(c2ncc(C)o2)C)cc1 CCCC(C#N)C(=O)NCC1(C(=O)N(C(C)CO)C)CC1 O=C(C1CCCc2scnc21)NC1(CCNC(c2cscn2)=O)CCC1 C1(NC(N(C)C(c2ccccc2)c2ccccc2)=S)CCN(OCC#N)CC1 C1(CCC(C)(C)NC(C(CC)NC(N)=O)=O)CCCCN1C(C1CCS(=O)CC1)=O c1(OCCC(=O)NC(CNC(CC2C(C)(C)C(O)C2)=O)(C)C)ccc(Cl)c(Cl)c1 C1(C(=O)NC(C(=O)N(C(CC(C)C)C)C)Cc2ccco2)CCCCC(=O)N1 C(C(CC(F)(F)F)NC(=O)CCCNCc1cccnc1)NC(C1C(C)C1C)=O C1(N(C(=O)COc2ccc(C)cc2)CC)CCOC(C)(C)C1 C1(N(C(=O)C(C2CCOCC2)O)C)CCN(C(=O)CNC(c2ccoc2)=O)CC1 C(C(F)C(=O)NCC1(O)CN(C(C2CCC2)=O)C1)NC(=O)OC(C)(C)C c1(C(=O)NCCNC(C2CCC(C#N)CC2)=O)cccc2ncsc12 C(CC(C(=O)N1CCC2CC12)NC(c1cn(C)nc1OC)=O)=CC C1(C(N(CCCNC(=O)C(C)(C)c2cscn2)C(C)C)=O)C(F)(F)C12CCC2 C(C(F)(F)C(C)(C)O)c1nc(-c2ncc(OC)nc2)nn1C1CCCC1 c1(NC(COCC(C)C)=O)cccnc1C(=O)NC(C)C(C)SC1CCCC1 C1(N(C(C=Cc2ncc(C)[nH]2)=O)C)CCN(C(=O)Cc2c[nH]nc2O)CC12CC2 N1(C(C2CC3(C(C(=O)OCC)C3)C2)=O)CCC2(O)CCCCC2(O)C1 C(=O)(C(C)NC(=O)C(C)N(C)C(C)=O)NCCOC CCC(CN=c1cc(NCCc2ncc[nH]2)nc(C)[nH]1)N(C)C Cc1cc(NC(C2C=CC(NC(C3CC(O)C3)=O)C2)=O)c(C)cc1O n1(CC)cnc2[nH]c(=NC(C)CC#N)[nH]c(=NC3CC4(COCCO4)C3)c12 N1(C(Cc2c(C)n[nH]c2C)=O)CCC2CN(C(=O)C(c3ccc(F)cc3)=O)C2C1 C=CCC(CC(C)C)C(=O)N1CCCC1Cn1cc(Cn2cnc(OC)c2)nn1 C(=O)(C1CCCc2ncnn21)N1CCC(COC)(NC(C2CC2(C)C)=O)CC1 C(CCCC(=O)NCc1cn(C2CN(C(=O)C(N3CCOCC3)C)C2)nn1)SC c1(C(=O)OC)c(Cc2cn(C3CN(C(=O)Sc4ccccc4)C3)nn2)noc1C CC(=O)CC(C)(C)C(=O)N(CCCn1cc(-c2cc(F)ccc2Cl)nn1)C N(C1COc2cccc(F)c21)C(=O)NC1C(C)(CC)C1 C1(C(C)(C)NC(CC2(NC(C)=O)CCC2)=O)CCCCN1C(=O)CC1(C)CCCC1 C(=O)(C(C(C)(C)C)c1cc[nH]n1)NC(CCNC(Cc1c(C)nsc1)=O)(C)C C1(C(=O)NC(CNC(c2c(C)ccc(C)n2)=O)(C)C)CN2CCC1(C)CC2 CCC(C)C(O)C(C)C(=O)NCCCN(C(=O)C(C)CC1CCC1)C CC1CCc2nc(NC(N3CCC(F)(F)CC3c3ccco3)=O)ncc2C1 C(=O)(CN=c1[nH]c2ccccc2s1)N1CC(CNC(CSC(C)C)=O)C2C1C2 c1(CNCc2cc(C(=O)Nc3cccc(OC)n3)cn2C)ccc(C)c(C#N)c1 C1(C(N(C2C=CC(NC(=O)CCCCCF)C2)C)=O)CC2(CCCCC2)C1 C1(CN(C(CCNC(=O)NC)=O)C)CCCCN1C(=O)C=Cc1ccncn1 c1(C(N2CC(c3n(CC)cnn3)C(CO)C2)=O)nc(C2CC2)ncc1Br Cc1c(F)ccc2[nH]c(C(N3CCCCC3C3CCCC3O)=O)cc12 CC(=O)C(C)CC(C)C(=O)NC(C(=O)NC1CC(=O)N(C)C1)C(C)(C)C C(c1cnc(C)s1)=CC(=O)NC(CN(C(c1cscc1Cl)=O)CC)C c1(C(C)C)cnnc(-c2nc(C3CCC(C(C)C)CC3)nn2C2CCC(C)C2)c1 C1(C(=O)NCCC2(CNC(=O)CNC(=O)NC3CC3)CC2)C2COCC12 C1(NC(c2cc(Br)cs2)=O)CN(c2ncnc3cc[nH]c23)CCC1(F)F N1(C(C(CC)(C)OC)=O)CC2CCN(C(C3(C(F)F)CCOCC3)=O)CC(C2)C1 C(C)(C)(CCCNC(c1cnc(C2CCOCC2)s1)=O)NC(C(C)C#N)=O C1(NC(C(c2c(OC)cccc2)O)=O)CC(C)CN(C(=O)Cc2cscn2)C1 C(CCS(C)(=O)=O)(C(=O)N1CCC(C)CC1CNC(c1cocn1)=O)OC c1(C(C)C)cccc(C(=O)NC(C2CCCN(Cc3cc[nH]c3)C2)C)c1 C1(CC(=O)NC(CC(=O)NCC2CC(C(=O)OC)C2)C)CC(C2CC2)C1 C#CC1(O)CCN(C(c2cc(C(C)C)nn2C)C(=O)NCCOC)C1 c1(C(C)C)ccc(C(CNC(C2(C)CCOC2)=O)NC(c2ccc(F)o2)=O)cc1 N1(C(c2ccc(F)c(Br)c2)=O)CC(C2CCN(C(C3(O)CCOCC3)=O)CC2)C1 Cc1cn2c(C(=O)NCCN(C(=O)CCC(F)F)C3CC3)c(C)nc2s1 C1(NC(CCC(=C)Br)=O)CC12CCN(C(=O)C(N1CCOC1=O)C)CC2 C(C(COC)C(=O)NC(C)CNC(c1cc(CS(C)(=O)=O)on1)=O)OC CC(CS(C)(=O)=O)C(=O)N1CCC2CN(C(=O)C3=CCCC3)C2C1 N1(C(C(C)SC)=O)CCC2CCN(C(C3CC(F)C3)=O)C2C1 c1(NC(CC2N(C(C3CCC(C(C)C)CC3)=O)CCOC2)=O)nc2c(s1)CCC2 c1(C(N(C)CC2CCN(C(c3ncn(C)n3)=O)C2)=O)cc(C(F)F)n(C)n1 N1(C(C)=O)CCCC(C2CCN(CC=CCCN(CC(F)(F)F)C)C2)C1 CCC(C)CC(C(=O)Nc1cncc(OC)c1)NC(=O)C1=CCCCO1 C1(O)(CNC(C(=Cc2ccccn2)C)=O)CCCN(C(=O)C(O)C2CC2)C1 C1(C(=O)NC(C)COCCO)(CC)CCCN(C(C2CN3CCC2CC3)=O)C1 C1(CCOC)CN(C(c2ccnnc2)=O)CCN1C(c1ccccn1)=O CN(C)S(=O)(=O)NCC(=O)NC1CCC1NC(c1cc(C2CCCC2)n(C)n1)=O CCC(CC)CCCC(=O)N1CCN(C(c2cccnc2NC)=O)CC1CO C1(NC(C2(c3ccccc3)CCCO2)=O)CCCCC1C(=O)NC1CC1 C12CC(C1(C)C)NC2=O.C(=O)(C(C)C(=O)OC)N1CC(=C)C1 c1(C(=O)NCC(CNC(CSCCC)=O)C)cc(OCC)cc(F)c1 CC1CN(C(=O)C2=CCCSC2)CCC1CNC(c1cnn2c1OCC2)=O Cn1ccc(C2(C(=O)NC3CC(NC(C4CCC4c4ccccc4)=O)C3)CC2)n1 C1(CC)CCC(C(=O)NC(C)CN(C(=O)CN(C2CC2)CC)C)CC1 N1(C(CC(C)C)=O)CCCC2CN(C(=O)CCCNC(N)=O)CCC12 c1(-c2cc(NC(C3(C)N(Cc4c(C)nns4)CC3)=O)on2)cccc(F)c1 C(=O)(C1=CCC(F)(F)CC1)NCC12CCC(NC(c3c(CC)ncs3)=O)(C1)CO2 C1(NC(c2cc3n(n2)CCO3)=O)C2CCN(C(=O)CCc3ccoc3)CC12 C(=O)(C1=C(C)OCC1)NC1CC(OCC(=O)N(CC#C)CCO)C1 N1(c2cc(NCC3(c4ccccc4)CCOC3)nc(C)n2)CCCC(N=[N+]=[N-])CC1 C1(C)(CC)CC(NC(c2ccc(Cl)cn2)=O)CN1C(c1cc(C)c(Cl)cn1)=O C1(C(N(CC(=O)NCC)C)=O)C2CCC(C2)N1C(C1CC12CCOCC2)=O N1(C(C2(OC)CCCC2)=O)CC23CCCC2(C1)CN(C(=O)CCC(C)N(C)C)C3 C(=O)(C(C)(C)C1=CCN(C(c2c[nH]nc2C)=O)C1)NCc1occ(C)n1 C(N=C(NC1CCc2nc(-c3cccs3)sc2C1)N1CCC(C)C(C)C1)SCC N1(C(COC)=O)CC(C)(C)C1C1CCN(C(c2sc(CC(C)C)nc2C)=O)CC1 C1(C(N2C(C)(CNC(C=CCN(CC)CC)=O)CCC2)=O)CCc2nncn2C1 C1(NC(c2ccc(O)nn2)=O)CC2CCC1CN(C(C13CCCC1C3(F)F)=O)C2 N1(C(c2c(CC)c[nH]c2)=O)CCC(NC(=O)Cc2ccc(F)cc2)C(CO)CC1 C1(NC(C(C(C)(C)C)O)=O)COC2C(NC(C3CN(C(N)=O)C3)=O)COC12 C=C(Cl)CCC(=O)NCC(C)(C)CN(C)C(C1CCCC1(F)F)=O N1(C(C2(CNC(C(C)SC)=O)CC2)=O)CC(C)OCC1C Cc1cc(C(=O)NC2CCCC2CC(=O)NCC(C)C(F)F)no1 N1(C(c2c(C=C)cnn2C)=O)CCN(C(=O)C(O)CC(C)(C)C)CC(C)(C)C1 c1(C(=O)NC(CNC(c2ncc(C)nc2)=O)C(C)C)ccc(C(F)F)c(Cl)c1 c1(OC)ccc(C)nc1C(N1CC(NC(c2cc(N)ccc2Cl)=O)CC1C)=O N1(C(c2cc(C)c(C(=O)O)o2)=O)CC(C2CCCN(C(=O)C(C)CO)C2)C1 C1(C(N(CC(CC)OC)C)=O)CN(C(c2cnc(C(C)C)[nH]2)=O)CC12CC2 N1(C(C2CC(C)N2C(=O)C=Cc2cncn2C)=O)CC2C(C1)C2(C)C CCC(C)(C)C(C)CC(=O)NCC(C1CC1)NC(c1ccn(CCO)c(=O)c1)=O C(CC(=O)NC(C)CC1CCC1)N(C)C(C1CCSC1)=O c1(C(=O)NC2(C)CCN(C(C(CCN(C)C)O)=O)C2)ccc2ccncc2c1 CC1CCC(Cl)=C(C(=O)N2CCN(C(C3CCC(=O)N3)=O)CC3(CC3)C2)C1 CC1CC(c2ccccc2)CCN1Cc1cn(-c2cccc(F)n2)nn1 C(=O)(CC(C)(O)CCC)N(CC(=O)NCCCCCC(C)C)CCC CC1CC(NC(=O)CN(C2CCCC2)CC2CC2)CCS1.C1(N)CC(NC)C1 c1(C(N(C2CCN(C(C(CN(C)C)O)=O)C2)C)=O)cc(F)c(F)cc1F N1(C(CCC(=C)Br)=O)CCN(C(=O)CCCCc2cnc[nH]2)C(CCO)C1 Cc1ccc(C(CNC(=O)CCC2CCCC2)NC(C2(Cl)CC2)=O)cc1 N1(C(c2c(C)nn(CCO)c2C)=O)CCC2(CC1)CC(F)CO2 N(C(=NCCCCl)NCC(c1ccc(Br)cc1)O)C1CCN(CCC)C1 c1(C(=O)OC)coc(C=CC(=O)NCC2CCCN2C(c2ccc(=O)oc2)=O)c1 c1(C(N2CCC(C)(NC(C(CCCC)O)=O)C2)=O)cc2cc([N+](=O)[O-])ccc2o1 CC1=C(C(=O)N2CCC(CNC(=O)C(C(C)C)c3cccc(Cl)c3)C2)CCO1 c1(OC)cc(C(N2CC(NC(=O)C(C(C)C)OC)C(C)C2)=O)ccc1Cl C1(CN(C(=O)COC)CC)CCCN1C1CCC1.c1(C=O)cc(CC(C)C)on1 C1(NC(=O)CCn2cc(COc3cccc(F)c3)nn2)(CO)CCC(O)CC1 C1(NC(c2cc(OC)c(Br)cn2)=O)CCN(C(=O)C(C)OC)C12CCC2 Cc1nc(N(C2CC(N)C2)C(=O)Cc2cc(Br)ccc2C)c2ccccc2n1 C1(NC(CC=CC=C)=O)CC2(CCC(CNC(=O)C(O)C(C)SC)CC2)C1 CC(C(C)(C)C(=O)NCC1(C)CC2CCC1C2)NC(C1CC2(CCC2)C1)=O c1(N2CCN(C(c3[nH]c(C)c(N)c3C)=O)CC2)ccc2c(c1)CCO2 c1(C(C)NC(=O)NC(COCCOC)C)cccc(N2CCCC2=O)c1 C1(=CCNC(CCSC)=O)CCN(C(c2cc(-c3cccnc3)nn2C)=O)CC1 C1(CC(=O)N(C2CCN(C(Cc3scc(C)c3)=O)C2)CCO)CCCCCO1 C1(NC(C(CNC(=O)C(C)(C)C(C)O)OC)=O)CCC(=O)N(C)C1=O C(=O)(C1CCCc2cnn(C)c21)N1CC(OC)C(OC(C)(C)C(=O)OC)CC1 c1ccsc1CN(C1CCCCC1)C.C(CC(O)c1cccs1)N C1(Nc2ncnc(CC)c2F)CCC2(C1)CN(C(C1CCC(O)CC1)=O)C2 N1(C(CS(=O)(=O)NC)=O)CCC(CNC(C2C3CN(C)CC23)=O)C(C)C1 C1(CN(C)C(C2CCCC23CC3)=O)CCCN(C(c2cccc(CF)c2)=O)C1 C1(C(=O)NC(C2CCN(C(=O)CCC3OCCO3)CC2)C)CCC(NC(N)=O)CC1 C(N=c1[nH]c(N2CC3CC3(CO)C2)nc2c1CCC2)C1(S(CC)(=O)=O)CC1 C1(=O)CCCCCN1CCCN(C)C.c1(CNC(=O)CC2CCCO2)ccccc1 c1(CNC(CCOCC)=O)cnn2c1CN(C(C1CC(C)CC(C)(C)C1)=O)CC2 c1(C(=O)NC(CC)(CNC(c2nc(Cl)cs2)=O)CC)cc2ccc(C)cc2o1 S(=O)(=O)(c1cc(C(=O)O)cs1)N1C(C(=O)OC)CCOCC1 O=C(C1CCCc2sccc21)NCCCC1(NC(C2CCOC2)=O)CC1 C1(C(=O)NCC#CCNC(c2c(C)[nH]cc2)=O)CCc2nnc(C)n2C1 Cc1c(N2CC(NC(c3ccc(C#N)cc3)=O)CCC2C)ncnc1C(F)(F)F CC(CCC(Cl)Cl)NC1CC2(C(=O)O)CC12 CC1CN(C)CCC1NC(=O)C#CCNC(c1cc(C#N)cs1)=O Nc1c(F)ccc(C(N2CC3(CCCC3NC(c3cn[nH]c3)=O)C2)=O)c1F c1(C(N(C2CCCN(C(=O)C3=CCSC3)C2)C)=O)ccc(C(F)F)c(F)c1 N#CC1(C(N2CCC(O)(CNC(=O)CCn3cncn3)C2)=O)CCOCC1 N1(C(COCCCC(C)C)=O)CCOC(CNC(c2cnc(CC(C)C)s2)=O)C1 c1(OC)cc(C)c(C(=O)NCCC2CCN(C(C3(O)CCC3)=O)CC2)c(C)c1 c1(C(=O)Nc2c(C)ncn2C)cc(F)c(Cl)cc1F CCCC(C)(CC)C(=O)N1CCC2C(C(=O)NC(c3ccncc3F)C)C2C1 CCCC(CC)CCC(=O)NC(c1c(C)cccc1Br)C(N1CC(C)CCCC1C)=O N1(C(C2CC(C)(CC)C2)=O)CCC=C(CNC(=O)CSc2nc[nH]n2)C1 c1(C(=O)NCC2(NC(C34COCC3C4)=O)CC2)cc(C(F)F)cc(F)c1 C(=O)(C1=CC2(CCOC2)C1)N1CCC(=CCNC(=O)C(F)C2CCC2)CC1 N1(C(C=CCOC)=O)CC(C(C(=O)NCC(F)Cl)OC)C1 O=C(C#CC1CCC1)NCC1CCCC(NC(C2(F)CC=CC2)=O)C1 S(=O)(=O)(c1cccnc1NCC1CCCOC1)NC(CC)CCOC C(CCCC(=O)N(CC(Cc1ccccc1)NC(C12CCC1C2)=O)C)SC C1(CN(C)C(C23CC(C(C)(C)C)(C2)C3)=O)CCCN1C(c1c[nH]c(=N)o1)=O N12CC3CC(C(C3)C1)Cn1cc(nn1)C2=O.C1(COCC(=O)NCO)CCCO1 CC1C(C)S(=O)(=O)CCN1C(C1CC(n2cc(-c3cncs3)nn2)C1)=O c1(NC(c2c(-c3ccc(N)cc3)n[nH]c2)=O)n[nH]c2cc(Cl)ccc12 C(Cc1ccccc1)(C(=O)N(CC(C)(C)C)CCC(=O)O)OC N1(C(C2C(C)(C)C2C#N)=O)CC2CCC1CN2C(C1CC1C(F)(F)F)=O CC1(C)CN(C(=O)CC2OCCO2)CCC1C(=O)NC(C(N)=O)C1CC1 N1(C(CCCC(C)NC(c2cc[nH]c2C2CC2)=O)=O)CCc2ccc(F)cc21 N1(C(C(CNC(c2ccnc(O)c2)=O)CC2CC2)=O)CCCCC12CC2 c1(NC(CN2C(C)(F)CCC2)=O)ccc(C2COc3ccccc32)cc1 C1(C(=O)NCc2c(C)nsc2C)CCN(C(=O)C(CC(C)C)N(C)C)CC1(C)C c1(C(c2nnnn2C2COC2)NCc2n(CC)nc(Br)n2)cc(C)cc(C)n1 CC1CC2CCC(C(=O)NCC(C(C)(C)C)NC(c3cc(Cl)c[nH]3)=O)CN2C1 N1(C(C(C)CO)=O)CCC(CNC(=O)Cc2nc3c([nH]2)CCCC3)C(F)(F)CC1 CC(CCNC(c1cc2ccncc2s1)=O)N=c1[nH]nc(-c2ccon2)s1 c1(OC)cc(C(C)NCc2ccccc2F)ccn1 c1(NC(c2cnccn2)C)ccc(S(=O)(=O)NCC2CCCO2)c2ccncc12 CCCC(C)(C)C(=O)NCCOCCC(=O)NCC1CCCC2(CC2)C1 N1(C(=O)C(C2CCC2)C2CCC2)CCC2CCN(C(=O)COC(F)(F)F)C2C1 c1(COC)nc(C)c(C(=O)NCC(F)CNC(=O)CC2CCOC2)s1 C(=O)(N=c1[nH]nc(CC)s1)NCC1CCN(C(CCCC)=O)C1 CC1CN(C(=O)C(C)(C)n2cccn2)CCC1N(C)C(c1coc(C(F)F)n1)=O c1(C(=O)NC(CC)C(=O)NCC2CCCCS2)ccc2c[nH]nc2c1 N1(C(C(C)=C(CC)C)=O)CC(CNC(c2c[nH]nc2C2CCCC2)=O)C(C)C1 Cc1cccc(CN2CCOCC(C(=O)OC(C)(C)C)C2)c1Br c1(-c2cn(C(C)C(=O)NCC(C3CCCC3)N(C)C)nn2)ccc(Cl)c(N)c1 C(N=c1nc2c(cnn2C)c(NCC2CCCCC2(F)F)[nH]1)C1CC(N(C)C)C1 c1(OC)ccc(Cl)c(F)c1C(N1CCN(C(C2CSC2)=O)C(C(F)F)C1)=O Cc1ncnc(NC(C)CCNC(c2ccccc2OC2CCC2)=O)c1Br N1(C(c2ccc(OCCOC)cc2)=O)C2CCC1C(NC(=O)C=CBr)C2 c1(OC)ccc(CNC(c2ccc(SC)o2)c2nnnn2C2CCC2)cc1C#N c1(NC(C2CN(C(c3ccc([N+](=O)[O-])o3)=O)CCC2O)=O)ccn2ncnc2c1 CC#CCCCC(=O)NCC1CC(C(N2CCOC3(CC3)C2)=O)CO1 c1(C(C)C(N2CCC(Cc3ccccc3Cl)C2)=O)cc2ccccc2s1 c1(C(=O)NC2CCN(C(C(CC)F)=O)C2)cn2c(n1)C(=O)N(C)CC2 N1(C(Cc2n[nH]c(=NC)s2)=O)CCC2C(C1)CN2C(C12CCC(C)(C1)OC2)=O CCC(CC)C(=O)N(C1CCC(CNC(=O)COCCCOC)CC1)C C1(NC(c2scc(CNC(C3CC(C)(CC)C3)=O)c2)=O)CCCCCC1CO CC1CC(NC(c2cccn(C)c2=O)=O)CCN1c1cc(C(N)=O)nc(Cl)n1 C(C(C)(CC)OC)N(C(CN(C(=O)CC1CC(=O)C1)CC)=O)C CN(C)S(=O)(=O)N(C)CC(=O)NC1(CNC(c2ccnc(C3CC3)c2)=O)CC1 N1(CC)CC(C(=O)NC2(c3ccccc3)CN(C(=O)C=C3CC3)C2)CC1=O C1(C(N2CCN(C(=O)C3CC3)C(CC(F)(F)F)C2)=O)CCC2(CCC2)O1 N(C(=NCCC)NCc1noc(-c2ccc(F)cc2F)n1)C(C#C)C(C)(C)C C=CCC(C(=O)NCCC(C)(O)CC)NC(c1ncccc1CC)=O N1(C(C(C)NS(CCC)(=O)=O)=O)CCC(NC(C2(OC(C)=O)CC2)=O)C(O)C1 CCCCCCC(C)CC(=O)N(CCCCCNC(c1cc(O)ncn1)=O)C CC(C(=O)NCCC1CN(C(=O)C2CC2)C1)OC1CCCC1.C12CC1NC2=O Cc1[nH]nc(C(=O)N(C)CCN(C(c2cnn(CCO)c2C)=O)C(C)C)c1C C(C)(C)(CCCNC(c1nc(OC)c(C)s1)=O)NC(C(CC)N(C)C)=O N1(C(C(n2cc(-c3cccc(OC)c3)nn2)C)=O)CC(SC)CC1(C)C c1(C(C)C(N2CC3(CCN3C(=O)C(C)C3(O)CCC3)C2)=O)ccc(S(C)(=O)=O)cc1 Cc1ccc(NC(C2CN(C(=O)C(C)NC=O)C(C)(C)C2)=O)c(CO)c1 c1(C(=O)NCC2NCC(OC)C2)nn(-c2ccc(C)cc2)c2c1CCCC2 N1(C(CN(CCCCCC)C)=O)CC2CC1(CNC(C1CN(C(N)=O)C1)=O)C2 C(c1ccc(F)cc1)=CC(N1CC=CC(NC(C2CCCCC2C(F)(F)F)=O)C1)=O N1(C(=O)OC(C)(C)C)CCOC(C(=O)Nc2ccc(-n3cc(Br)cn3)nn2)C1 c1(C(=O)NCC2CCN2C(=O)CC2C=CCC2)cnc(C2CC2)nc1O Cc1ccc2n[nH]cc2c1C(=O)NC(C)CC(C)NC(c1ccc(=N)[nH]c1)=O C1(CNC(C2(COCC)CC2)=O)CCCC(N(C)C(c2sccc2F)=O)C1 C(=O)(C1CCCc2nncn21)NC1C(NC(c2c(C)nc(C(F)(F)F)s2)=O)CC1 c1(NC(C(N2C(CC)CC(O)C2)c2cc(Cl)n(C)n2)=O)cccc(Cl)c1C c1(C(N(CCC(C)NC(C2CCC2n2cccn2)=O)C)=O)cc(Cl)cc(F)c1N c1(C(=O)NC2CCC(C(N(CCCC(=O)N(C)C)C)=O)C2)nccc2cc[nH]c12 C(=O)(C(O)C(C(C)C)OCC)N(C1CCCN(C(C(C(=O)OCC)F)=O)C1)CC c1(CC)cccnc1C(=O)NCC(C)(C)CN(C(=O)CC1CC2CC2C1)C c1(NCCCn2c(C)ncc2)nc2ccccc2nc1N1CC=C(Br)CC1 C1(CC(=O)N(C)CC2N(C(c3scc(OC)c3)=O)CCC2)CC2CCC(C1)N2C CC(C)CCC(C(=O)NCCC1(C)CC1(F)F)NC(C1CCC(C(N)=O)C1)=O c1(SC)nc(C(=O)NCCC2CCN(C(=O)C(N)=O)C(C)C2)c2ccccn12 Cc1cc(C)c(C(=O)NC2CC3(CCN(C(=O)CC4CCC4(F)F)C3)C2)c(C)c1 Cc1cc(C(=O)NC2CC(O)CN(C(c3ncoc3C)=O)C2)cnc1C C(C)(C(O)C(C)C)NC(CN(CCOC)C(c1coc(C(F)F)c1)=O)=O c1(OCC)ncc(C(=O)NCC(C)NC(c2ncoc2C(C)C)=O)cn1 N1(Cc2cc(C(=O)OCC)n[nH]2)CC(O)Cc2cccc(Cl)c21 CC(C)C(CC(=O)N1CCOC2CC12)NC(=O)C=C1CCOCC1 N1(C(CCOCCN(C(=O)CCN(C)CCO)C)=O)CCC(CCCO)C1 C(=O)(C(C)(C)CN(C)C)NC(CN(C(=O)CCCc1nncn1C)CC)C c1(CNC(C(=O)Nc2ccc(OCC(=O)NC)c(Cl)c2)=O)n[nH]c2c1CCCC2 C1(NC(C2N(C)CCC2)=O)CCC2CC1CN2c1nc(CC2CC2)ns1 C1(F)(CNC(c2ncoc2-c2ccco2)=O)CCC(CNC(C2CC23CC3)=O)C1 c1(N2CC(F)(C(=O)Nc3c(OC)nn(C)c3)C2)ncnc2ccc(I)cc12 CCC(CC)CCCC(=O)N1CCC2(CC2C(=O)Nc2cnc(O)c(C)c2)C1 C=C(C)CN=C(NCC(Cc1ccccc1)C(F)(F)F)NCC1(CO)CC(C)C1 O=C(C1=NN(c2cccc(Cl)c2)C(=O)CC1)c1noc(C2CC2)n1 C(=O)(C(C)CC(F)(F)F)NCC1(CNC(C2CN(C(C)C)C2)=O)CC12CCC2 CCCCC(CC)CCC(=O)NCC(C)CNC(C1CCC2(CCC2)C1)=O c1(CC(=O)NCC(CN(C(Cc2c(C)n[nH]c2)=O)C)C)cncc(Br)c1 c1(C(C)C)cncc(C(C(=O)NC(C)(C)C)N(C(CF)CF)C)c1 c1(C(N2C3C(CNC(c4c(COC)cc[nH]4)=O)C(C3)C2)=O)ccnc2c1CCO2 C=CC(C)(O)CC(=O)NCC1C(C)CCCN1C(c1ccccc1OC)=O c1(NS(CC(C)C)(=O)=O)ccc(S(=O)(=O)NCCNC2(C)CCC2)cn1 N1(C(c2cc(C(C)C)on2)=O)CCN(C(c2cc(CF)on2)=O)CC(C)(F)C1 c1(C(N2CC(CC)N(C(=O)C3=CC(C)(C)C3)CC2)=O)cc(S(N)(=O)=O)sc1C c1(C(=O)NCC(CC)NC(=O)C(C)OCC(F)(F)F)cc(OC)nc(Cl)c1 c1(OC)ccc(-n2nc(C3CCC(C)CC3)nc2CC2CC2(F)F)cc1 N#CC1(C(=O)NCC2CCCN(C(=O)CCC3CC3(F)F)C2)CC2CCC1CC2 Cc1c(F)cc(C(N2C3CCC2CN(C(C2(CC4CC4)CC2)=O)C3)=O)c(F)c1N c1(OCC(=O)Nc2nc(C)oc2C)ccc(Br)c(Cl)c1 n1(CC(=O)NC2C(NC(Cc3n(C)nnc3)=O)C2)cccc(C(F)(F)F)c1=O CC(CC(=O)NCC1(NC(=O)CC2CC(C)(C)OC2=O)CC(F)(F)C1)C(F)F C12(C(C)C)CCC(NC3(C)C(C(=O)NC(C4CC5(CCC5)C4)CO)CCC3)C1C2 c1(C(C)C)ccc(=NC(=O)N(C)Cc2cc(F)cc(F)c2Br)[nH]n1 N1(C(C2(CC(C)C)CCNC2=O)=O)CCCCC(NC(c2ccnnc2Cl)=O)C1 N1(C(CC(=C)C)=O)CCN(C(=O)CC2COC(C)(C)CO2)CC1CCOC N1(C(C(CC#C)C2CC2)=O)CC(C(N2CCC(C)(C)C2)=O)CC12CCC2 N1(C(C=CC(=O)OCC)=O)CC(CNC(=O)COCc2cccs2)(CO)C1 N1(C(C2C(C)=C2)=O)CC(C)CN(C(c2c(C)ccc3n[nH]cc23)=O)CC1C N1(C(C2CCCC(NC(C=C(CCC)C)=O)C2)=O)CCC(C(N)=O)C(C)(C)C1 C(=O)(C(C#N)C(C)(C)C)N1CCCCC(CCC(=O)NCc2nc(C)oc2)C1 C(=O)(C1=NOC(C)(C)C1)N1C(CNC(COCCSC)=O)CC(O)C1 C#CCCN=c1scc(-c2ccc(Cl)s2)n1C1CCC(N(C)C)CC1 C1(O)(CNC(C(=O)Nc2ccc(C(C)(O)C(F)(F)F)cc2)=O)CCCNCC1 CCC(C)C(CC(=O)NCC1(CC)CCCCO1)NC(=O)Cn1cncn1 c1(C(C)NCc2cn(CC3CCC(=O)O3)nn2)c(F)cccc1Br c1(C(=O)NC2CN(C(=O)CC3(O)CCC3)CCC2F)c[nH]c2nccc(Cl)c12 c1(OC)cc(Br)cnc1C(N1CC(NC(=O)C(O)CN(C)C)CC1CO)=O CCCC(C(=O)NC1CC(CNC(c2cnoc2-c2ccccc2F)=O)C1)OC C=CCCC(C(=O)OCC)N(CC(=O)OC(C)(C)C)CC C1(CC)CN(C(=O)COCCCn2ccnn2)CCN1C(=O)Cc1nccn1C c1(CC(=O)NCC2CC(COC)CN2C(C2CCOC2)=O)cc(C)cc(F)c1 C1(NC(c2c(CC)scn2)=O)CC2CC1N(C(c1cc(C(C)=O)cs1)=O)C2 c1(OCC)cc(C=CC(=O)NC2CCCC2C)ccc1OCC#N c1(NC)cnc(C(C)C)nc1C(=O)NCC(C(C)(C)C)NC(=O)CC1CC=CC1 CCC1=NOC(C(=O)NCC2CCC(C(=O)NCc3cccnc3OC)CC2)C1 C(=O)(C(F)(F)C(C)O)NC1C(CN(C(C(n2cnc(C#N)n2)CC)=O)C)CCC1 CC1=NS(=O)(=O)NC=C1C(=O)NC(C)C(C)(C)NC(=O)C#CC(C)C N1(C(C2COCC(C)O2)=O)CCC2CC2(C(=O)NCc2ncccn2)CC1 CC(C)C(CNC(=O)COCC1CCCO1)NC(C1CCCCO1)=O C(=O)(C1CN(c2snc3ccccc23)c2ccc(OCO)cc21)OC C(=O)(CCCCCn1cc(C(C)O)nn1)N1CC(C(C(=O)OCC)C)C1 N#CC1CCCC(CC(=O)NC2CC2C(=O)NC2CCOCC2)C1 N1(C(c2c(C)scc2)=O)CCC2(NC(C3CC3C3CCCCC3)=O)CCCC12 C=CC1(C(=O)NC(C2CCCC2O)C)CCN(C(C2COCC(C)O2)=O)CC1 c1(C(=O)NC2C(CNC(c3csc(C(F)(F)F)c3)=O)C2)cn2ccnc2cn1 N1(C(C(CC(C)C)C)=O)CCc2[nH]nc(CNC(C3(N4CCOCC4)CC3)=O)c2C1 Cc1ccc(C(=O)NC2CC3CN(C(c4cc(CF)on4)=O)CC23)cc1[N+](=O)[O-] c1(C(=O)NCC(CNC(C(CSC)C)=O)CO)cc2c(nn1)CCC2 CC1CCN(CC2CC(N(C34CC(F)(C3)C4)C(C3CCN3)=O)C2)CC1C1CCCO1 CC1(C)CC(NC(C2CCS(=O)(=O)C2)=O)CN(C(=O)Cc2ccc(F)c(F)c2)C1 C12(CNC(c3cc(C)oc(=O)c3)=O)CC3CC(CC(C3)C1N)C2 c1(C(N(C2CCN(C(=O)COC3CCC(C)CC3)C2)CC)=O)ccnc(O)c1 C1(NC(C2(CC(=O)N(CC(N)=O)CC(N)=O)CC2)=O)CCC2(CC2)C1 N1(C(c2[nH]c(=NC)sc2)=O)CC2(C1)CN(C(c1ccccc1C(C)(C)C)=O)C2 c1(C(=O)NC2C3(CC(NC(CN(C)CC)=O)C3)C2)nccc(C#N)c1F c1(CNC(C(C)SC)=O)ocnc1C(=O)NC1CC(=C2CC2)C1 N1(C(C)=O)CCCC(C(=O)NC(C)(C)CN(C)C(c2csc(Cl)c2Cl)=O)C1 c1(C(=O)NC2CC3(CC(NC(C(C(C)C)C)=O)C3)C2)ccc(C#N)nc1O N1(C(COCCCCCC)=O)CC(NC(c2ccc(CN(C)C)nc2)=O)C(O)C1 C(=O)(CC(C)(C1CCC1)C1CCC1)NCCCN(CCCNC(COCC)=O)C C1(C(=O)NC(CC=CC)C(=O)NCC[Si](C)(C)C)CC(C2CC2)=NO1 O=C(C1=NN2CCCN=C2N1)NCCC1CCCN(C(=O)C2=C(Cl)CC2)C1 C1(CC=C)(C(=O)NCC2(CO)CC(C)C2)CN(C(=O)C(C)N(CC)CC)C1 CCCC(O)C(=O)NC(CNC(c1[nH]cc(C(C)=O)c1C)=O)C(C)(C)C C1(C(N(C(C)CCNC(=O)C(F)(F)C(F)F)C)=O)CNC(=O)C(C)(C)C1 CCC(C)C(O)C(=O)NC1(CNC(c2cccc(CF)c2)=O)CCOCC1 N1(C(CC2CCCN(C(C(CC(C)C)O)=O)C2)=O)CCOC2(CCC2)C1 C(=O)(CC1CNc2ccccc21)N1CCC(C(C)NC(C=CSC)=O)CC1 C(=O)(CC1=CCOCC1)NCC12C(CN(C(c3cc(CC)nc(O)c3)=O)C1)C2 C=CC(C)(CCOC)C(=O)NCC#CC(=O)NCc1sc(C)cc1C C(C(O)CC(=O)N1CCCC1CN(C)C(c1ccncc1C(=O)OC)=O)N(C)C N1(CC(=O)NCCOCC)CCCC(C)(CNC(=O)Cc2ccc(C)o2)C1 N1(C(CCCOCCC)=O)CCC(CNC(=O)CC2CCSCC2)C(CC)C1 C(=O)(C(F)CCC(C)C)N1CCC(CC(=O)NC2(CC)CCOCC2)CC1 c1(C(=O)NCC23CC(CN2C(C2(C(N(C)C)=O)CC2)=O)C3)cc(C#N)ccn1 CC(C)CC(CCc1ccccc1)C(=O)NCC(CNC(=O)C(C)(Cl)Cl)CO C1(F)(C(N2CCC(N(C(=O)C(C)c3ccco3)CCC)CC2)=O)CCN(C)CC1 N1(C(C=Cc2ccc(C)s2)=O)CC(NC(C2CCC(C)(C)OC2)=O)CC(C)C1 c1(C(N2CC(CCCNC(c3c(CC)noc3)=O)OCC2)=O)ccc(F)cc1O N1(C(C2C(C#C)C2(C)C)=O)CC2CCN(C(c3cc(F)ccc3N)=O)CC2C1 c1(C(N(C)CC=CC(=O)NCC2COCCO2)=O)cccc(CO)c1 C1(C(N2CCC(C(=O)OC)C2)=O)C2CC(O)C(C2)N1C(=O)C1=CC2C=CC1C2 c1(C(=O)NCCn2c(C)ncc2)cc2cccc(-c3ccc(B(O)O)cc3)c2[nH]1 N1(C(C2=CC(C)(CC)C2)=O)C2CCCC1CN(C(=O)C=CC=C(Cl)Cl)C2 C1(C#N)(NCC(CC2CCCO2)N(C)C)CCN(C(=O)OC(C)(C)C)C1 Cc1ccc(O)cc1NC(=O)C(CC1CCCC1)NC(=O)CCc1cnn[nH]1 [N-]=[N+]=NCCCCC(=O)N1CC=CC1Cn1cc(CC(CO)CO)nn1 c1(C(=O)NCC2(O)CCCN(C(c3nc(Cl)cs3)=O)C2)ccc2n[nH]cc2c1 Cn1cc(Cl)cc1C(N1CC(CNC(C2CC(=C3CCC3)C2)=O)C(O)C1)=O Cc1c(N)cc(C(N2CC(C(C)NC(c3occc3F)=O)C2)=O)cc1[N+](=O)[O-] c1(C(=O)NC2C3CN(C(c4c(C)ccnc4)=O)C(C3)C2)sc2ncccc2c1Cl C(=O)(C1(C)CCCc2ccccc21)NC1CN(C(c2cc(C)[nH]c2C)=O)CC1C C(N=c1ccnc(Cl)[nH]1)C1C(NC(c2cc(Cl)ncc2F)=O)CCC1 N1(C(CN(C)C(c2ccsc2)=O)=O)CCN(C(C2CCNC2=O)=O)CC1CF N1(C(C(CC)(C)F)=O)CC2CC(C)N(C(c3cccc4ncnn34)=O)C2C1 CN=c1[nH]cc(C(=O)NCC2CN(C(=O)C3=CCC3)CC2C)o1 CCCC(CC(=O)NC1CN(C)CCC1O)NC(=O)Cn1cccnc1=O CC1(C)COC(C(=O)NC2CC(CC(=O)NC3CC3O)C2)C1 C1(NC(c2cc(SC)c(C)o2)=O)CC(F)CN(C(c2nnc(C(C)(C)C)s2)=O)C1 C1(CC(=O)NC)CN(C(=O)Cc2cn(C)cn2)CCN1C(=O)C1=CCC1 Cc1nn[nH]c1C(N1CC(O)(C(C)NC(c2cn(CCF)nn2)=O)C1)=O c1(C(N2CC(CCC)C(NC(C3NC(=O)OC3C)=O)C2)=O)cnc2n1CCCC2 C1(NC(COCC(=C)C)=O)CC2CC1N(C(=O)C(c1cccnc1)OC)C2 c1(C(N)=O)sccc1CNC(C(C1CCN(C(C2(N(C)C)CCOC2)=O)C1)C)=O C=C(C)C1OCCCC1C(=O)NCC1CCCCN(C(c2cnnc(C)c2)=O)C1 C(=O)(CS(=O)(=O)CC(C)C)NC1C2CN(C(Cc3ccc(C)c(C)c3)=O)CC1C2 C(=O)(CCCCCSC)NCC(C)(C)NC(C1CC1C1CCCO1)=O C=CC1(CC(=O)NCCOC)CN(C(=O)C(CO)c2ccccc2)C1 C1(CNC(COC(CC)(C)C)=O)CN(C(c2nc[nH]n2)=O)CC1C C1(C(=O)NCCc2cc[nH]n2)CN(C(=O)CCC2CC2(F)F)CC12CCC2 C(CCC(=O)NCC1(C)CCCO1)N(C(=O)C=Cc1ccco1)C C(=O)(C(C(C)C)NC(C)=O)NCCCCNC(c1ccc(COC)o1)=O CCCS(=O)(=O)CC(=O)NCC1(F)CC(NC(=O)CC(C)(C)O)C1 C(CN=c1[nH]c(=NCC(C)(C)COCC(F)F)[nH]c2ccccc12)OC(C)(C)C C(=O)(C(Cn1cccn1)NC(=O)C(C)=C1CCC1)N(CCC#C)C N1(C(C2CCOC3(CCC3)C2)=O)CCc2nncn2CC1 N1(Cc2ncc(OC)nc2)CCC(F)(F)C(C(=O)NC2CCNC2=O)C1 c1(C(N2CCC3C(C2)CN3C(=O)CC23CCCC2C3)=O)ccc2c[nH]nc2n1 N#Cc1ccc(CNC(=O)C(c2cccs2)NC(c2cccnc2)=O)o1 N1(CCSC)C(=O)NC(c2cc(Cl)cnc2Br)C2=C1C(C)N(C(C)(C)C)C2=O C1(C(=O)Nc2cc(Br)ccc2N2CCOCC2)COc2cc(Cl)ccc2O1 c1(C(N2CCC(C)(NC(C(C)C3CCC3)=O)C2)=O)c[nH]c2ccc(Cl)cc2c1=O c1(CN(c2ccnc(NCC3=CCCCC3)n2)C)ccc(F)c(Br)c1 N1(C(c2cn3c(n2)CCC3)=O)CCCN(C(C2CC23CCOCC3)=O)C(CO)C1 c1(C(CCN(CCc2cn(CC(=O)O)nn2)CC)(F)F)cccc(C)c1 Cc1ccc2c(c1)CC(C(N1C3CCC1CN(C(=O)CCCCC#N)C3)=O)O2 c1(C(N2CCCC(C)(CNC(C3(O)CCSC3)=O)C2)=O)cnc2ncc(Cl)cn12 c1(C(=O)NC(C)(C)CNC(c2ccn(CC(F)(F)F)n2)=O)cnc2[nH]cncc1-2 c1(C(=O)NC2CC(CNC(C3(CC#C)CCCOC3)=O)C2)cc(C)cc(F)c1 c1(C(c2n(CCOC)nnn2)NCc2ncc(Br)s2)sc(Br)nc1Cl c1(OC)cc(C(=O)NCC2CN(c3cc(O)ncn3)CCO2)ccc1C#N C(=O)(N=c1cc(C(F)(F)F)[nH][nH]1)C1CCN(C(c2ccc(C)cc2Cl)=O)C1 N1(C(c2c[nH]c(=NC)s2)=O)CCN(C(=O)CNC(N2CCCC2)=O)C(CF)C1 CC1(C)CCC(C)(C(=O)NC2CC3(NC(c4cnsc4)=O)COC2C3)CC1 c1(CNC2(c3n(C4CCC(C(=O)OC)C4)nnn3)CCSC2)cc2occc2s1 C(=O)(C(C(C)(C)C)OC)OC.c12cn(cn1)CCn1ccnc1C(OC)OC2=O CC1(C)COCC1CC(=O)NCC1CC(CNC(=O)C=Cc2cccnc2)C1 C1(CNC(c2cc(CC)[nH]n2)=O)CCN(C(=O)C(C)C#N)CC1C1CC1 c1(C(=O)NC2CCC(CCNC(C(C)SCC)=O)C2)cccc2c1CCCCC2 c1(C(=O)NCC(C2N(C(CCC)=O)CCC2)(C)C)cnc(OC(F)F)c(C)c1 C(=O)(C(O)CC(F)(F)F)NCc1ccc(C(=O)NC(CSC)(C)CO)cc1 N1(C(c2cc(C)n(CC)c2C)=O)CCC(C2CCN(C(=O)CSC)CC2)CC1 C1(C(=O)OC)CCC2(CCC2)N1CCC1(C(=O)O)CCOC1 c1(C(=O)NC(C(O)CO)C2CC2)coc2c1CN(C(C13CCC(CC1)C3)=O)C2 c1(NC(c2ccc(N3CCC(N)CC3)nc2)=O)cc2ccccc2nc1Cl N1(C(c2c(OC)cnnc2)=O)CCOCCC1C(=O)NC1(c2ccsc2)CC1 Cc1c(Cl)ccc(C(=O)NCC2CC(O)(CNC(C3C(C)(C)C3(C)C)=O)C2)c1O CC1(C)CN(C(C2(CF)CC(F)(F)C2)=O)CC1CNC(=O)Cn1cccnc1=O c1(C(N2C(CNC(c3c(C)cc(Cl)cc3)=O)CC2)=O)cc(S(=O)(=O)N(C)C)c[nH]1 Cc1c(C(=O)NC2C3CN(C(=O)CCc4ccccn4)CC23)cccc1Br c1(C(=O)NC2C(NC(c3ccc(C)o3)=O)CC2)c(C2CC2)noc1C C1(CC)CN(c2ncncc2C)CCN1C(=O)C(C)(C)C#N Cc1nn(C)c2ccc(C(=O)NC3CC(NC(=O)CC#N)C34CCC4)cc12 c1(C(N2C(C(N(C)Cc3cccc(C)c3)=O)CCCC2)=O)ccc2ocnc2c1 c1(CN(CC(=O)O)C(C2CC(F)(F)CO2)=O)ccc(Cl)cc1 CC1(C)CN(C(C2CN(S(N)(=O)=O)C2)=O)CC2(CN(C(C3CCCC3)=O)C2)O1 N1(C(c2cc(C#N)sc2)=O)CCCC(CNC(C2CC2C2CC2)=O)CC1 C(N=c1[nH]cc2ncnc-2[nH]1)C1C(NC(C(CC)(C)CC)=O)CCCC1 c1(C(=O)NC(C(C)NC(c2n(OC)cnc2C)=O)C(C)C)cnn2cccnc12 N1(C(c2cc(CCC)c(C)s2)=O)CCCC(NC(=O)CC2SC(=N)NC2=O)CC1 C1(OCC)CN(C(=O)C(C)n2cncn2)CC1CNC(c1cc(C)sc1C)=O C12(CC(=O)NCC(c3cccs3)O)CCC1CN(C(=O)Cc1ccccn1)C2 C1(C(=O)NCCc2cn(-c3cc(C(=O)OC)ncc3)nn2)CCC12CCOCC2 N1(C(COCCN(C)C)=O)CC2(CC(NC(=O)C=CC3CCCCCC3)CO2)C1 C12(NC(C(C)N(C)C)=O)CCCC(NC(c3ccc(SC(F)F)cc3)=O)(C1)C2 S(=O)(=O)(c1ccc2[nH]c(=NCC3CC4C=CC3C4)sc2c1)NC(C)(C)COC(F)F c1(C(N2C(COC)(CNC(=O)C3=NOCC3)CCC2)=O)cccc(C2CC2)c1Cl C1(NC(c2csc(O)n2)=O)CCSC12CN(C(c1ccc(O)cc1)=O)C2 CC(c1ccsc1)=CC(=O)NC(C)(C)CN(C(=O)CC1CC2CC2C1)C c1(-n2ccc(C(=O)NC(C(C)NC(C(C)=CC)=O)C)n2)cc(F)cc(F)c1 c1(C(=O)NC(CC=C)C)cccc(CNC(=O)CN(C2CCCC2)C)n1 c1(Cn2c(COCC)ncc2)c(Br)cc(C(=O)O)n1C CCCC(C)CC(=O)NCC(C1CCNCC1)F C1(NC(c2ccc(C#N)cc2)=O)CN(C(c2sccc2F)=O)C2(CCOCC2)C1 c1(C(c2n(CCC)nnn2)NCC(=O)NC2(C)CCOC2)ccc(OCC)cc1 N1(C(c2nnn(CC)c2C)=O)CC(CCNC(C2CC(F)(F)CS2)=O)OC(C)C1 C1(O)(C(=O)OC)CCN(CC2(Cc3ccc(O)cc3)CCCC2)CC1 c1(C(N(C)CC2(O)CCCN(C(C(C)C3CC3)=O)C2)=O)ccc2c(n1)CCCC2 C1(NC(C2C(C)C2)=O)C2CCC1CN(C(C1(F)CC=CCC1)=O)C2 C=CCC(CC=C)C(=O)NCC1CN(C(=O)CN(C)C(N)=O)CCO1 C(=O)(C1=CCCOCC1)N1C(C(=O)NC(CC#C)C(=O)OC)CC(C)CC1 C1(CC(=O)NCC(CCCC)NC(=O)CCc2nc(C)cs2)CC(O)C12CCC2 C(CCCCCNC(C1(F)CC=CC1)=O)N(C(=O)CC1CCOC1)C N1(C(C(C)OCC#C)=O)CCC(C)N(C(c2cn(CC(N)=O)nn2)=O)CC1 C1(NC(CCSC)=O)CCN(C(=O)CCc2ccc(F)cc2Cl)C(C)C1 CCCC(C(=O)NC1CCC1)NC(C1(C)COC(=O)N1)=O CCCC(CCC)CC(=O)NC1CCCC1NC(=O)CC1CCC(=O)O1 Cc1cc(C(N2CCOCC(C(=O)NCC(O)CNC(N)=O)C2)=O)c(C)n1C N1(C(CC(C)OC)=O)CCC2(CC1)CC(CNC(=O)C1CCc3c[nH]nc31)C2 c1(N2CC(NC(c3cccc(O)c3O)=O)C(O)C2)ncnc2n[nH]c(I)c12 C1(C(=O)NCCN(C)C(C2(c3nc[nH]n3)CC2)=O)CC2CCC2C1 N12CC=CC(C1)C2=O.N1(CC(=O)Nc2cn(CC=C)nc2)CCN(C)CC1 C1(C)(CNC(C(C(C)(C)O)F)=O)CC(F)(F)CN1C(=O)Cn1nc(O)ccc1=O N1(C(C(CCOC)C)=O)CCC(C)(C)C(CNC(C2(O)CCCCC2)=O)C1 C1(C(N(C(CC)CC)C)=O)CC(O)C(O)CC1CNC(=O)C(C)CC1CCCC1 C1(C(=O)NCc2nc(COC)sc2)CCCCC1NC(=O)C(C)OCC(C)C c1(N2CCC(O)(C(=O)NCCCSC)C2)nc(C2CC2)nc2ccccc12 CC1CCC(C)(C(=O)NC(C)C(CO)NC(c2scnc2C2CC2)=O)CC1 c1(CCC(N2CCCC(N(C(c3cnsn3)=O)CC)C2)=O)ccc2[nH]ccc2c1 c1(CC)c(C(c2nnnn2C(C)(C)C)NC2CC2c2ccccc2F)ccn1C n1(CC(=O)NC23CC(CNC(CC(C)C)=O)(OC2)C3)nnc2ccccc2c1=O c1(OC)cc(C(N2CCC(C3CCN(C(=O)C4=NNC(=O)C4)C3)CC2)=O)cc(Cl)n1 c1(C(C(=O)NC(C)C(=O)Cc2ccccc2)(F)F)ccc(F)cc1F C1(CNC(C(C)NC(COC)=O)=O)CCC2(CCN(C(=O)CC=C(C)C)CC2)O1 Nc1c(C(N2CCCCC2CNC(=O)C=Cc2cnc[nH]2)=O)sc2ncccc12 C(=O)(C(C)C(C)S(C)(=O)=O)NC(C(C)C)CNC(C1(C)CCC1)=O N1(CC(CNC(c2cc3c(cc2)C(C)(C)C=C3)=O)F)C(=O)c2ccccc2C1=O C1(CNC(C2C(CCC)C2)=O)CN(C(c2ccc3ccoc3c2)=O)CC(C)(C)O1 Cn1nc(C(=O)NC(CNC(=O)Cc2ccc(O)cc2)C2CC2)cc1F c1(C(=O)NCC(C2CCOC2)NC(=O)Cc2cscn2)cnn2c1CCC2 c1(N(C)Cc2c(C)n[nH]c2)cc(NC(C2CCCO2)C)nc(C(F)(F)F)n1 c1(C(=O)NCC2CC(NC(C3OCCC(C)C3)=O)C2)nnn2c1CSCC2 C#Cc1ccc(C(=O)NCC(CO)NC(c2ccn(C3CC3(F)F)n2)=O)cn1 C1(C(N(CC(C)NC(C2(O)CCSC2)=O)C)=O)CC(C)(C)OC(C)(C)C1 Cc1c(C(=O)NCC23CC2CN(C(c2cc(C4CC4)nn2C)=O)C3)ncn1C CC1CC2CCC(C1)N2C(C1(C(C)NC(c2ccc(O)cc2)=O)CC1)=O C(c1ccc(C)c(C)c1)=CC(=O)NCC1CCC(NC(c2cnc(OC)s2)=O)C1 C(=O)(CS(=O)(=O)CCCc1ccccc1)NC1(CO)CN(C(C(CC=C)C)=O)C1 C1(C)(CCC)CCCN(c2cc(NC(C)CCn3cncn3)nc(C)n2)C1 C(C)(C)(CCCC(=O)NOCCCC1CC1)NC(c1ccn(C(C)C)n1)=O C1(C(=O)NCC(=O)NCC#C)C2CCCC2CN1C(=O)C(C)NC=O c1(C(N2CC(NC(COC3CCN(C)CC3)=O)C2)=O)cccc2ccsc12 C(C)(CCC(=O)N1CCCC(CN(C(=O)CCc2ccc(F)nc2)C)C1)SC C(CS(=O)(=O)CCNC(c1ncc(I)s1)c1nnnn1-c1ccc(Cl)cc1F)OC N(C1c2ccccc2CC1NC(=O)C(C)c1ccsc1)c1nc(C)cc(C)n1 N1(C(C2C=C(C)CS2)=O)CC=CCC1C(=O)N(CC(O)C1CC1)C C1(CC=C)(NC(=O)CC(C)(F)F)CCN(C(C2CC3CC2CC3O)=O)CC1 N1(C(CCC(=O)NCC)=O)CC2CCC(C1)N2C(=O)C(CC)CC(F)F C1(F)(C(=O)NCCC=CC=C)CCN(C(=O)C(CC)SC)CC1 c1(CN2C(CNC(Cc3c(C)[nH]nc3Br)=O)CC2)ccc2nonc2c1 NS(=O)(=O)CC(=O)N1CC(CO)(NC(=O)C=CC(F)(F)F)C1 N(C(=NCCC(C)SC)NCc1ccccc1OC)Cc1nc(CC)oc1 c1(C(=O)OCCNC(=O)NCCCOCCC(C)(C)C)ccc(O)cc1 S(=O)(=O)(c1ccc(N2CC3CCC(C2)O3)c2cnccc12)NCCC#N Cc1csc(=O)n1CCC(=O)NC1CN(C(=O)C(C)N(C)C)CC1C CCC(CC(F)F)C(=O)NC1(C)CN(C(c2ccc(OC(F)F)c(Cl)c2)=O)C1 N1(C(c2nn(CC)c(O)c2)=O)CC2(C1)CN(C(C1CC1(C(C)C)CC)=O)C2 C1(CC=C)(NC(=O)CCCCOC)CCCN(C(c2cc(C)n(CC)c2C)=O)C1 C1(NC(c2c(C(=O)OC)n(C)nc2)=O)CC(CNC(=O)C(C)(F)F)C12CCC2 N1(C(C(c2ccccc2)C)=O)CCCC(C(N2CC(CO)C(O)C2)=O)CC1 C1(C(N2CCC(CC=C)(NC(c3ccc(C)o3)=O)C2)=O)CC2CC1CC2(F)F C1(NC(C(CO)NC(c2cccc3c(Br)coc23)=O)=O)CCCC23OCCC2CC13 CC1CC(NC(c2nnc(S)n2C)=O)CN(C(c2ccn(C)c(=O)c2)=O)C1 c1(C(N(CC(CC)NC(c2conc2C(C)C)=O)C)=O)ccc(OC)cc1C c1(C(CNC(COCCCC#C)=O)NC(=O)C(C)CC2CC2)ccccc1F C1(CC(C)C)COCCN(c2cc(N(C)CCC3CC3)ncn2)C1 c1(C(=O)NCCNC(=O)C(C2CCCO2)NCCC)ccc(COC)cc1 c1(OCC)c(CN(CCC(C)C)C2CC2)cc(Cl)cc1Br c1(CNC(C2CC23CCNC3)=O)c(F)cccc1Br C(=O)(CC(C)CCC=CC)N1CC(Cc2ccc(-c3cn(CC)nn3)cc2F)C1 C1(C(=O)N(CCO)Cc2ccccc2)CC(=O)N(CCOCC2C3COCC23)C1 N1(C(c2c[nH]c(=N)s2)=O)CC2(CC2)CC1CNC(=O)C=Cc1ncc[nH]1 CC(C)(CC(=O)NC1CCC1NC(c1cc[nH]c1)=O)C(F)F C[S+](C)CCC(O)C(=O)N(C1CCN(C(C2(C)COC2)=O)C1)CCO Cc1nc(-c2ncccn2)sc1C(=O)NC12CC(C1)N(C(C1COC(=O)C1)=O)C2 c1(C(C(=O)NC2CC2)N(CC=C)Cc2cccs2)nc(Br)ccc1OC C1(C)(NC(c2c(CC(N)=O)occ2)=O)CCN(C(c2snc(O)c2Cl)=O)C1 Cc1cccc(CC(N2CCC2CNC(c2cnc(C3CCC3)s2)=O)=O)c1 c1(C(=O)NCC(CC)NC(C2COC(C)C2)=O)cc(F)cc(N)c1N c1(CC(=O)N(C)CC2CCN(C(CS(CC)=O)=O)C2)ccc(OC)c(C(C)=O)c1 C1(OC)CC2CC(C(=O)NCC3CCN3C(=O)C(C)(C)c3cc[nH]n3)CC12 N1(C(c2ccc(C)cn2)=O)CC(C)C(C)(CNC(c2cc3occc3s2)=O)C1 c1(C(N(C(C)CNC(=O)C=CC2CCCC2)C)=O)ccnc2ncccc12 c1(OC)cccc(CC(=O)NC(C)CC2CN(C(=O)C(C)(C)N(C)C)C2)c1 C1(NC(c2c(CCC)n[nH]c2)=O)CN(C(=O)C=Cc2c[nH]nc2C)CC12CC2 C1(C)(CCC)CCN(C(=O)C(CCOCCO)NC(C2COCCC2C)=O)C1 N1(C(c2[nH]cc(C)c2C)=O)CCN(C(=O)NC(=O)C(Cl)(Cl)Cl)C2(CC2)C1 N1(c2ccc(C(=O)OC)cc2)CCN(C(C2CC3(CCC3)C2O)=O)S1(=O)=O C1(C(N(CCCCNC(C(C)(C)OCC)=O)C)=O)CCc2ncnn2C1 Cc1cc(=NCC2(C(N)=O)CCC2)[nH]c(=NCCn2ccnc2C)[nH]1 N1(CCC(=O)NC2CCCC2NC(=O)C=CCN2CCCC2)CCCCC1 CCCC(O)(CNC1CCCC1CCC(C)C)C(F)(F)F Cc1cc(F)cc(CN2CCC(C(=O)Nc3ccc(F)cc3O)C2)c1O C12(NC(c3cc(C)cc(N)c3)=O)CCCC1CN(C(=O)Cn1c(C)csc1=O)C2 N1(C(C=C(C)Cl)=O)CCC2(CCC2)C(NC(=O)C(CCC(N)=O)NC(C)=O)C1 CC12CCN(CC1)CC2C(=O)NC1(CNC(=O)Cc2cnccc2Cl)CCOC1 c1(C(=O)NC(CC=C)C(=O)N2CCOC(CC(C)C)C2)c[nH]c2ccncc12 c1(CCCC(=O)NCC(CCOC)NC(=O)C(C)C2CCC2)ccc(F)cc1 O=C1NC2CN(C(c3cscc3C(F)F)=O)CC2NC1=O N1(C(c2c(OC)scc2)=O)CC(OC)CC1NC(=O)COCCCF N1(C(c2n(CC)ncc2)=O)CCC(NC(=O)COCCN(C)C)C1C1CC1 N1(C(CC(C)SC)=O)CCC(C)(C)C(C(=O)NCC2CCC3(CC3)C2)C1 Cc1nc(Cl)[nH]c(=NC2CC(NC(=O)NC(=O)CCSC(F)(F)F)C2(C)C)c1F C(=O)(CS(=O)(=O)N1CC(O)CC1C(N1CCCCC1C(N)=O)=O)OCC N1(C(C(CCC)C)=O)CCC2C(CCN2C(c2ncc(Cl)cn2)=O)C1 Cc1ccc(CC(=O)NC2CC2NC(c2cc(C(F)(F)F)cs2)=O)o1 CC(=O)CCCC(C)C(=O)NC(C(=O)Nc1cnc(C)nc1)c1ccoc1 c1(NC(=O)CCn2ccc(C(F)(F)F)n2)ccccc1.C1(=O)C(C)N1.CC(=O)O.C(C)=O N1(C(C(=Cc2cnc[nH]2)C)=O)CCCC(C2(NC(C3CSCCS3)=O)CC2)C1 c1(C(=O)NCCCc2c(C)cccc2Cl)nc2n(c1Cl)CCCC2 C1(C(NOCC=C(C)C)=O)CC(O)CCN1C(C1COCC(C)O1)=O Cc1nc(Cl)ccc1CC(N1CCCC(NC(C23CC(F)C2C3)=O)C1)=O CC12CC(C(=O)NC3CC(NC(=O)C(C)(C)c4ccccc4)CC3O)(CCO1)C2 c1(C(N(CC(C)NC(=O)CC2CC2C)C)=O)nc(Cl)ccc1N c1(NC)cccc(C(N2CCC(CF)(NC(c3ccc[n+]([O-])c3)=O)C2)=O)n1 c1(OCC(=O)NC2CC2CNC(c2cccnc2)=O)ccccc1 CCC(C#N)(CC)C(=O)N1CCC(O)C(NC(=O)CC(O)c2ccccc2)C1 N1(C(C(c2ccccc2)NC(=O)CC(O)C2CC2)=O)CCc2sccc2C1 Cc1cc(C(N2CCCCC2CN(C(=O)C(O)C(C)(C)C)C)=O)cnc1C(F)F C12(C(N(CCCCC)C)=O)CCC(CN(C(C3(O)CCSC3)=O)C1)C2 C1(C(N(CCCN(C(CCN(CCC)C)=O)C)C)=O)CCCC1O C1(OC)CC(C(=O)NC(=O)CC2C=CCCC2)CN(Cc2ccc(F)cc2C)C1 N1(C(C(C)(C)NC(CN2CCC(C)CC2)=O)=O)CCCC(C#N)C1 C1(C2CCN(C(C3C(C#N)C3(C)C)=O)CC2)(NC(c2c(C)nco2)=O)CC1 c1(C(=O)NCC(CNC(CCCOC)=O)(C)O)cc(Cl)c(F)cc1[N+](=O)[O-] CCC(CCC(=O)NC1CC2CCC1N2C(c1csnc1C)=O)OC C1(C(N2CC(CC(C)NC(=O)C(O)C3CC3)C2)=O)C2CCC1(C)C2(C)C CC1(C)CCCC1CN1CCC(C)(c2ccccc2)C1.C12CCC(C1)CC(=O)N2 Cc1c(F)ccc(C(=O)NC2CCN(C(=O)C3=CCCS3)CC2(C)C)c1N c1(C(N2CCC(NC(CC=CC=C)=O)C(F)C2)=O)n[nH]c2ccc(O)cc12 CCCC(C)(C)CC(=O)NC1CCCC(C(=O)NCCCCCCC(C)C)CC1 c1(C(=O)NCC2C(NC(CN3C(C)CCCC3)=O)COC2)cncc2ccsc12 c1(NC(=O)NCCOCCOC)nc(C)cc(=NC2CCCC2C(C)OC)[nH]1 CC1CCC(C)(C(=O)N(C2CN(C(=O)CNCCS(=O)(=O)COC(C)C)C2)C)C1 C1(NC(C(C)C(C)(C)C)=O)CCC12CCN(C(c1ccc3cnnn3c1)=O)CC2 Cc1cccc2c1CC(C(=O)NC1(C)CCCN(C(=O)C=CCF)C1)O2 C1(NC(C=C(CC)CC)=O)CN(C(=O)CCC(=O)NC2CCCC2)CCC1F c1(N2CCCC(C(C)NC(CSCC)=O)CC2)nc(SC)nc2ccccc12 C(=O)(C1=CC2(CCN(CCONC(=O)CN3CCN(C)CC3)C2)C1)OC N1(C(CCCC(C)(C)NC(C2CC3CCC3C2)=O)=O)CCC(C2CCOC2)C1 C(=O)(C1=NOC2CCCC12)NC(CC)C(=O)c1ccccc1 C(=O)(C1CCCn2cnnc21)NCCC1CN(C(C(c2cccc(C)c2)=O)=O)C1 N1(C(CCCC(C)=O)=O)CCN(C(c2cc(OC)c(Cl)s2)=O)CC(CO)C1 C1(CNC(C2(CC)CCC2)=O)C2CCCC1N(C(=O)Cn1nc(C)c(Cl)c1C)C2 c1(C(=O)NCCN(CCCC)C)nc(CNC(=O)CC2CC(F)(F)C2)oc1C C1(C(c2nnnn2CC(F)F)NC(C2(CO)CC2)C)C2(CCC2)C12CCC2 C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CCN(C(CC(C=C)C)=O)CC12CCC2 N1(C(CCCCC#C)=O)CCOCC(C)(CNC(=O)C2=CCC2)C1 C1(CNC(C(C(=C)C)(C)C)=O)CC2COCC2N1C(C12CCC1CC2COC)=O C1(CCOC)(NC(=O)CC2CC(C)C2)CCN(C(C2CCCC(F)(F)C2)=O)CC1 C(CC(C(=O)NCC1CCCC1NC(C1CC1C)=O)NC(C)=O)SC C(=O)(C(C)C(O)CC(C)C)NC1(CF)CN(C(C2=C(C)CCC2)=O)C1 c1(COC)nc(N(C)CC2(F)COC2)cc(N2CCC(C)(N3CCCC3)CC2)n1 c1(CCC)nnc(S)n1CC(=O)NCC1CCN1C(=O)C=Cc1cnc[nH]1 C1(NC(CC2N(C(C3CC(CC)C3)=O)CCCC2)=O)CC2CC1C(O)C2O c1(C(N2CC(NC(c3ccoc3)=O)C3(C2)CC3)=O)ccnc2cc(F)cnc12 c1(C(N2CCN(C(C(CCC)(C)CC)=O)C(C)C2)=O)cccc2c1CCC(=O)N2 c1(OCC)ccc(CC(=O)NCC(C(C)(C)C)NC(c2occc2CC)=O)cc1 Oc1cc(CCn2cc(-c3c(Cl)cncc3Cl)nn2)ccc1Br c1(OCC(=O)N(C)CCNC(=O)CCCn2cncn2)ccc(Br)cc1 C1(C(=O)NCC(=O)N(CC)CC)CC(F)(F)CN1C(=O)CCOC(C)=O.C(CF)O C1(CN(c2ccnc(NCCc3nnc(Br)n3C)n2)C)CCCC(O)C1 c1(OC)ccccc1-n1cnc(C(=O)NCC(F)CNC(=O)C(C)C(F)F)c1 N1(C(=O)Nc2c(Cl)cc(C(F)(F)F)cc2Cl)CCc2sc(-c3csc(C)c3)cc2C1 N1(C(CC(C)C2CC2)=O)CC2(CCN(C(=O)CC3COC(C)(C)CO3)C2)C1 C1(CNC(C(C#C)(C)C)=O)CN(C(c2[nH]c(O)nc2C)=O)CC1(C)C C1(NC(c2cn(CC=C)nc2)=O)CCCCN(C(=O)CCc2nnc(C)n2C)C1 C1(NC(C(C)=CC)=O)CN(C(C2C3CCC4C(C3)CC24)=O)Cc2nccn2C1 C1(c2cn(C)nc2)CCCN1N1CCC(CC(=O)NCC(C)(C)C(C)(C)C)C1 C1(O)(C(=O)NCC2N(C(C(C(C)C)N3CCCC3=O)=O)CC2)CCCC(C)(C)C1 CCC(CC)C(C)C(=O)N(C1CCCCC1NC(c1occ2c1CCOC2)=O)C C1(CNC(=O)C(C2CCN(C(=O)CN3CCCC3=O)C2)F)(CO)CC2(CCC2)C1 C1(NC(C(C(C)O)(C)C)=O)CCCCCCC1NC(=O)C=C1CCCCC1 c12ccc(cc1)s2.C(=O)(C(COC(C)(C)C)C1CCC1)NS(CC)(=O)=O c1(C(N2CCC(CCOC)CC2)=O)cccc(-c2cn(C(C)C(=O)O)nn2)c1Cl c12ccc3ccc(nc3c1)C(=O)CC1CN(C(=O)CO1)C2=O.CC(=O)OC(C)=O N1(C(c2c(NCC)ccc(C)c2)=O)C2CCCC1CN(C(=O)CC1CC1C)C2 CC1CN(C(=O)CC(CNC(=O)Cn2cncn2)C2CCC2)Cc2nncn21 N1(C(c2c(OC)ccs2)=O)CC2(CCC(NC(=O)C(C3CCC3)OC)CC2)C1 c1(C(=O)NCC2CC(NC(C3C(C)(C(F)(F)F)C3)=O)C2)ccc(F)cc1[N+](=O)[O-] C1(CNC(c2c(C(C)C)scn2)=O)CCCCN1C(=O)CC1CCCC12CC2 C#CC1(O)CC(C(=O)NC(C2CCCCN2C(=O)Cc2cnnn2C)C)C1 C(=O)(N=c1cc(Cl)n(C)[nH]1)c1nc(NC(COC)=O)sc1 c1(C(N2CC(NC(c3c(C)[nH]nc3Cl)=O)C(C)CC2)=O)cncc(N=[N+]=[N-])c1 Cc1n[nH]cc1CC(=O)NC1(C(=O)NC(c2nnnn2C)C)CCSC1 c1(C(=O)NC2(CC=C)CCN(C(=O)C=CCO)C2)cc(F)c(Cl)c([N+](=O)[O-])c1 C(C(=O)N1CC=CC1COC)(C(C)(C)C)NC(c1c(CC)occ1)=O C(=O)(C1CNC(=O)c2ccnn21)N1CC(NC(CCCC(C)(C)C#N)=O)C1 S(=O)(=O)(c1ccc(Cl)c(C(=O)O)c1)N1CCN(C(c2nn(CC)nc2C)=O)CC1 c1(OC)c(C(N2CCCN(C(C3CC(C)C3)=O)CC2C)=O)ccc2c1CCC2 c1(C(N2CC(O)(c3cn(CC4CCCO4)nn3)C2)=O)c(F)cccc1Cl c1(C(CNC(C=C(COC)C)=O)NC(c2cscc2F)=O)ccc(F)cc1F c1(C(=O)N(C2(CN3CCCCC3)COC2)CC2CCCCC2)ccnc(CO)c1 C(C)(CC(=O)NC12CC(NC(=O)CCc3csc(C)n3)(C1)C2)OC N1(C(c2c(C)nc(CO)o2)=O)CCOCC(F)(CNC(=O)C(F)OC(F)(F)F)C1 c1(N(C)CC2CC(C)CC(C)C2)nc(N(C)Cc2nccn2C)c2c(n1)CCS2 C(=O)(C(C)(C)CF)N1C(CN(C)C(C2CC2C(F)(F)F)=O)CCC1 Cc1ccc(C(=O)NC23CC(NC(C4CC45CCCOC5)=O)(C2)C3)c(N)c1F c1(C(N2CC(C3CN(C(c4c(C)n(C)cn4)=O)C3)C2)=O)cccc2ncc(C)n12 c1(C(=O)NC(CN(C(=O)CN2CCCC2=O)CC)C)cc(C(F)(F)F)cn1C N1(C(CC(=O)NCC)=O)CCCC2CN(C(c3cnc(OC)cn3)=O)CCCC12 N1(C(Cn2ccc(=NC(=O)C3CN(C(N)=O)C3)[nH]2)=O)CCC2(CC1)CC2CO Nc1nc(Cl)cc(Cl)c1C(N1CCC(NC(=O)C(F)=CCCF)C(CO)C1)=O C1(CCCC)CN(C(c2c(C)nn(C)c2F)=O)CCN1C(=O)C=CC(=O)OC C(=O)(CCCCCN(C(=O)Cn1c(C)ccc1C)C)N1CC(NC(CC)=O)C1 C1(C2CN(C(c3cc(C(N)=O)cn3C)=O)C2)(NC(CC2N(C)CCCC2)=O)CC1 CC1CN(C(=O)CC(O)CNC(=O)C=CC2CCCCC2)CCCO1 n1(CCCOC)nnnc1C(c1nc(C)no1)(C)NC(COC)C1CC1 C(CCC(C)C(=O)NCCc1ccc(CNC(=O)C=Cc2ccco2)cc1)OC C1(OC)CC(CNC(C2CN(C)C(=O)N2)=O)N(C(=O)C=Cc2cc[nH]c2)C1 N1(CC#C)CCN(C(C23CC(CO)(CN2C(=O)C2=C(Cl)CC2)C3)=O)CC1=O C1(n2cc(C(CC)(C)C)nn2)CCCN(C(=O)CC2C=CCC2)C1 CCC(CCC(=O)N1CCC(C(O)CNC(=O)Cc2ccn(C)c2)CC1)OC CS(=O)(=O)c1cccc(CN2CCC(F)(CNC(=O)CC3CC3)C2)c1 CCCC(CCC)C(=O)NC(C)(CNC(=O)CCCC1CCCO1)CC C(=O)(C(CNC(C1CC2(CCO1)CC2)=O)C(C)(C)C)NCCC(C=C)(C)C c1(C(N2CCC(NC(c3c(C)ncnc3)=O)C2)=O)ccc2scc(Br)c2c1 c1(C(N(CC(CNC(CC2C(C)=NNC2=O)=O)O)C)=O)c2ccccc2nn1C c1(C(=O)NC(C)CN(C(=O)CNS(=O)(=O)C2CC2)C)cc(C#N)c[nH]1 C1(C)(C(=O)OC)CC(OC)CN1C(=O)NC(C1CCCCC1)CCO.C(C)(C)(C)O N1(C(c2c(C)cc(OC(C)C(=O)O)nc2)=O)CCC2(CC1)NC(=O)NC2=O c1(C(C2C=CC2)NCCCOCC2CCC2)nnnn1C1CCOC1 N1(C(CCSCCC)=O)CCN(C)C(CNC(c2cccc(C(=O)NC)n2)=O)C1 CCC(C)(C)CC(=O)NCC(CCNC(=O)CCC(C)N(C)C)OC Cc1ccccc1-c1nc(C(N2CC3(NC(c4cnoc4C)=O)CC2C3)=O)cs1 c1(C(N(C(CNC(C2(CC(=O)OC)CC2)=O)C)CC2CC2)=O)oc(C2CC2)nc1C c1(C(N2C(C(=O)Nc3c(CC(=O)OC)cccc3)CC(O)C2)=O)cccc(F)c1Cl N1(C(c2cncc(N)n2)=O)CCN(C(c2cc3n(c2)CCCC3)=O)CC12CC2 C(CC(C)(C)C)(C(=O)N1CCC(N(C)C(c2ccc(F)cc2Cl)=O)C1)OC CC1CCN(C(c2c(Cl)cnn2C)=O)C(CNC(c2ccnn2C(C)(C)C)=O)C1 CC(C)C(C(=O)NCCCNC(C1CCCC2CC12)=O)NS(C)(=O)=O C1(C(N2CCN(c3c(C#N)scc3)CC2)=O)COC2(COC2)C1 C12(CCNC(=O)CCc3ccccn3)CCC(C1)N(C(=O)C1=CCCS1)C2 c1(N2CCC(N(CCC)C(c3cncc(Cl)c3)=O)C2)cc(C2CC2)nc(Cl)n1 C1(NC(CN(C(C(C(C)C)SCC)=O)CCOC)=O)CC(C)CC(C)(C)C1 c1(C(N2CC(N(C(C(c3ccc(C)cc3)O)=O)C)C2)=O)cc(C)cc2c1CCC2 N1(C(c2sncc2C)C(=O)NC(CC)(C)C)CCN2CCC1C2 C1(NC(C(Cc2cn[nH]c2)NC(c2c(C)cn(C)n2)=O)=O)CCC(N=[N+]=[N-])CC1 C1(OC)CN(C(=O)CNC=O)C(C)(CNC(c2ccsc2C#N)=O)C1 C1(C(=O)N=CCN(C(=O)CCC2CC2)CCC)OC2CCC1C2 c1(C(C)CC(=O)N(CCCCNC(=O)C(C)(C)c2cccs2)C)ccccc1F CN1CCC(CNS(=O)(=O)CCC2CCCO2)CC1=O c1(C(=O)NC2CN(C(C=CC(CC)=CC)=O)CC2C)cccc2c1OCC(=O)N2 c1(CNC(C(n2cc(-c3cncc(OC)c3)nn2)C)=O)ccnc2c1CCCC2 c1(CNC2C(C(=O)NC(c3ccncc3)C)C2)ccccc1Cl C(=O)(C1=C(Cl)CCOC1)NCCC(C)CCNC(=O)CNC(c1cccs1)=O c1(C(N(CCN(C)C)C)=O)ccc(-c2nc(C3CCC(F)C3)n(C3CC3)n2)cc1 c1(OC)cc(C(N2CCCC2CCC(=O)Nc2cnc(Br)c(C)n2)=O)cc(C)c1 CC(C)CC(C(=O)NC1CCN(C(c2nccc(CO)n2)=O)C1)c1ccccc1 N#Cc1ccoc1S(=O)(=O)N1CCCC1CNc1ccc2[nH]ccc2c1 C1(c2n(CC=C)nnn2)(NCc2nc(CC)cs2)COCCC1C N1(C(c2ccc(COC)[nH]2)=O)CCC2(CC1)CN(C(=O)C(C)(C)C1CCCC1)C2 c1(OC(C(=O)NCCN(CCOC)C)(C)C)cccc(COC(C)C)c1 c1(C(N2C3C(NC(CCc4scc(C)n4)=O)C(C3)C2)=O)ccn2cnnc2c1 CC(C)C(C)(O)C(=O)NC1CC(CNC(=O)COc2ccc(Cl)c(F)c2)CC1O C1(CNC(CCc2ccc(C)o2)=O)CN(C(=O)CC(O)CN(C)C)CC1C c1(NCC2CC(C)N(C(c3coc4c3CSC4)=O)C2)cnc2ccccc2n1 c1(C(N2CC=C(CNC(CC3C(OC)CC3)=O)CC2)=O)nccc2cccnc12 N1(CC)CC(C(N2CCC(NC(C3(C(F)F)CCCCC3)=O)CC2)=O)CC1=O C(C(C)(C)C(=O)N1CC(F)(CNC(=O)CC2CCOC2C)C1)NC(C)=O c1cncn1C.C(C(=O)NCC1(C(C)NC(=O)C2CC2)CC1)OCCOC Cc1cc(C(=O)NC2(CF)CN(C(c3cc4n(n3)CCCC4)=O)C2)c(N)c(C)c1 c1(CC)ncc(C(N2CC(CNC(c3oc(C)cc3C)=O)CC2C)=O)c(O)n1 C1(C(N(CC)CC)=O)CCCC1NC(C1CCCN1C(C)C)=O C1(C(N2CCC(N(C(=O)C(C)=C3CCC3)CC)C2)=O)CC2(C1)CC1(CCC1)C2 Cc1cccnc1CC(N1CCCC1(C)CNC(=O)CC1CCOCC1)=O C12(CNC(C(C)NC(=O)NC)=O)CC1CN(C(c1cc(C)[nH]c1C)=O)C2 c1(C(N2CCN(C(c3c(C)snc3)=O)C3C2C3)=O)cccc(S(=O)(=O)NC(C)C)c1 C1(C(N2C(C)CN(C(C(CCC=C)(F)F)=O)C(C)C2)=O)COc2ccccc2C1 C1(CNC(c2cncnc2)=O)CN(C(C2CCC3CCC2O3)=O)CC2(CCC2)O1 CC1=C(C(=O)NC(C)CCN(C(=O)C(O)CCc2ccccc2)C)CCCC1 n1(CCC(=O)N(CC(C)NC(c2cnc(Cl)s2)=O)CC)cnc(C)cc1=O C1(CNC(CC=CCC)=O)(NC(c2ccnnc2C)=O)CCCCC1C c1(C(=O)OC)cc(C(=O)N(CCNC(=O)C(F)=C(C)C2CC2)C2CC2)c(F)cn1 c1(C(N2CC(CNC(C(C)C#N)=O)C(C)(C)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 CC(CC(=O)N1C2CCC(C2)C1CC(N1CC(CCO)(CO)C1)=O)C(F)(F)F N1(C(C=CCC)=O)CCC2CCN(c3nc4ccc(OC)cc4s3)CC2C1 C1(CNC(C(C)C)=O)CN(C(c2c(O)ccc(F)c2Br)=O)CCC1(F)F O=C(C1=NOC2COCC12)NCCN(C(=O)Cc1cccnc1F)C1CC1 CCCCCCC(CC)C(=O)NCCN(C1CCCCC1)C(=O)CCC1CCC1 C=CC(C(=O)NCC1(F)CN(C(C2CC2C(C)(F)F)=O)C1)OC c1(CC(=O)NCC(C2CCC2)NC(CCCSC)=O)csc2nccn12 C(=O)(CC1=CCCCC1)NCc1nc(C(N2CC(C)(C)OCC2)=O)c(C)o1 C1(C(N(CCNC(c2ccc(SC)s2)=O)CCOCCO)=O)CC2(CCC2O)C1 c1(C(N2CC(C)C(CNC(c3nncs3)=O)CC2)=O)cc(Cl)cc(Cl)c1F c1(OCC)ccc(C(=O)NCc2ccc(NCC3CC(F)(F)C3)cc2)c(CO)c1 c1(COC)cccc(C(F)(F)F)c1.c12ccc(cc1)SCC(=O)N1CC(C1)N2 C(=O)(C(C)(C(F)F)c1ccccc1)NCC(CNC(COCC(=O)NC)=O)(C)O N1(C(C2(C(=O)OCC)CC2)=O)CC2(CCCCC2)C1.C12C(C1(C)C)C(=O)NC2 CCC(CC)C(=O)N1CCOCC1CCNC(=O)CC1CCCC(C)O1 C1(C(N2C(CNC(C3(C)CC(=C)C3)=O)CC(OC)C2)=O)CC(=O)N(C)C(=O)N1 N1(C(C2C(NC(C(COC)N(C)C)=O)CCCCC2)=O)CCCC2(CCCO2)C1 C1(CNC(C(C2CCCSC2)N(C)CCOC2CC2)=O)CCSCC1 N1(C(CC(C(=O)NC)N)=O)CC2CC1(CO)CN2C N1(C(c2cc[nH]c2)=O)CC2CCN(C(c3cccc(Br)c3F)=O)C2C1 N1(C(c2c(OC)cccn2)=O)CC(C(=O)Nc2cc(C)cc(Br)c2)CC(F)C1 CC1C(NC(C23CC(C(F)F)(CO2)C3)=O)CCCN1C(=O)CNc1nccs1 C1(NC(C2CCN(CC)C2)=O)CC2CC1CN(C(c1nn(C)cc1[N+](=O)[O-])=O)C2 c1(C(=O)NCC(CC)(C)NC(=O)CCCCSC)cc2c(C)cc(C)nc2s1 CC1(C)C(NC(=O)CSC(F)F)CC1CC(N1CCC(Oc2nccs2)CC1)=O Cc1cc(C(=O)N(C(C)Cn2ncc3ccccc23)C)cc(C)c1C#N c1(C(=O)OC)nn(C)cc1C(=O)NC1CCN(C(=O)CCOc2cccnc2)C1 CCCC(C(=O)N(C(CNC(=O)C=NOC)C1CC1)C)OC c1(C(N2CCC(CNC(C3C4CC5C(C4=O)C35)=O)C2)=O)cn2ccsc2n1 C1(C(=O)NC2CCC(NC(=O)CCn3ccnc3C)C2)(OC)CCCOC1 C1(C(N(CCCCCNC(CCN(CC(C(C)C)C)C)=O)C)=O)CC2CCC1O2 C1(C(N2CCC(N(CCCC)C(c3cnco3)=O)CC2)=O)CCC2CC1CO2 c1(C(N2CCC(CC)(NC(C3CC3F)=O)CC2)=O)ccc2c(c1)CCCS2(=O)=O C(C#Cc1cccnc1)NC(C1(SC)CN(C(c2ccc(C=C)cc2)=O)C1)=O C1(CNC(C2(C=C)CC2)=O)COCCN(C(c2cc(C#N)oc2C)=O)C1 c1(C(NC(C2N(C(C(CC=CC)CC)=O)CC2)=O)=O)ccnc(P(C)(C)=O)c1 c1(C(N2C(CNC(=O)CSCC#N)CCC(C)C2)=O)nn(C)c2ccc(F)cc12 c1(NC(=O)NCC(=O)NC2CC(O)C(O)C2)c(F)cccc1Cl C1(c2n(C)ccn2)CN(C(C2(C)CC=CCC2)=O)CC1NC(c1cccnc1)=O C(CSC)(CN=c1cc[nH]cc1S(=O)(=O)N(C)CC1CC(C)(C)CO1)OC CCCS(=O)(=O)C(C)C(=O)N(C1CN(C(=O)CN2CCN(S(C)(=O)=O)CC2)C1)C Cc1cnn(C)c1C(=O)NC1CC2(C1)CC2NC(c1ccc(F)s1)=O C1(C(N2CCC(C(C(N)=O)O)CC2)=O)C2CC3C(C2OCc2ccccc2)C13 Cc1ccc(F)c(NC(c2ccc(CNC(=O)C#CC(C)(C)C)s2)=O)c1 CN1CCC(C)(C(=O)NCC2CCCN2C(c2cc(C(N)=O)[nH]n2)=O)C1 c1(NC(=O)NC(C=C)Cc2ccc(F)cc2)ccc(F)c(F)c1Cl CC1OCC2(CCNCC2)C1N(C(=O)C(F)(F)C(F)(F)F)c1cccc(Br)c1O c1(CC)ccc(NC(=O)C(F)(F)F)cc1S(=O)(=O)C(=O)Nn1c(C)nnc1C CC1(C(=O)NC2CCCC2NC(C2CCCN2C2CCOCC2)=O)CC=CCO1 C1(C2CCCC2)(C(N(C)CC2N(C(C(OC)OC)=O)CCC2)=O)CCNC1=O C1(NC(C(N2CCSCC2)C)=O)CCCC(NC(C23CC(CCO2)C3)=O)CC1 c1(NC(=O)NC(C)C)ccc(C(=O)NC(C)CN(C(=O)C(C)C(C)O)C)cc1 C1(NC(C(CC)OC2CCCC2)=O)C2CC1CN(C(=O)CC1CC=CCC1)C2 c1(CC(C)C)cc(C(=O)NCC2CCN2C(=O)CC(O)c2ccccc2)n(C)n1 c1(OC)ccccc1C=CC(=O)NC(C)(CNC(C1CC1C(C)O)=O)C1CC1 N(C(=NC1CCC1)N1CCOCC2(C1)CC2(F)F)C1CCC(C(=O)OC)C1 C1(C)(COC)CC(NC(=O)CC2(C(F)(F)F)CC2)CN1C(=O)CSC(F)(F)F Cc1cc(F)c(N)cc1C(N1CCCC(NC(c2nccc(Cl)c2C)=O)CC1)=O N1(C(c2c(C)cnnc2)=O)CCC(C)(C)C(NC(C2CC(C)(C(C)(C)C)C2)=O)C1 CC(C(=O)NC1CCCC(C(N2CC(C)(C)C2)=O)CC1)S(C)(=O)=O C(=O)(C1=CCN(C(c2cccc(C)c2C)=O)CC1)NC(C#CCCC)(C)C CCC(C(=O)NCC1CCN(C(=O)CCNC(=O)Cn2cnnn2)C1)SC c1(C(=O)NCC(CNC(COCCCOC)=O)F)cn(C(C)(C)C)nc1C CCCC(C)(O)C(=O)N(CC(O)CN(C)C(c1ccc(NC(C)=O)cc1Cl)=O)C CCCCC(C)(F)C(=O)NC1CC(NC(c2cc(O)nc(N(C)C)n2)=O)C(O)C1 N1(C(c2c(OC)cc(Cl)cc2)=O)CCN(C(=O)C(C)n2cccc2)CC(C)(C)C1 S(=O)(=O)(C1=Cc2ccccc2OC1)N(C)Cc1nc(C2CCCCC2)cs1 C1(CC(=O)NCC2CCCN2c2nnc(C(F)F)o2)CCC=CCC1 C(=O)(N(CCO)OC)C1(C)N(C(C2C(OCC)CC2)=O)CC=C1 C1(C(=O)NCC(N(C(CSCC#C)=O)C)C2CC2)CCC1(C)C c1(OC)cc(C(N2CCOC(C(C)NC(C3C=C3C)=O)C2)=O)ccc1C#N c1(C(=O)NCC(C)N(C(C(COCc2ccccc2)OC)=O)C)ncc(C)cn1 Cc1cnn(CCCNC(=O)C#CCNC(=O)C(C)Cn2cccn2)c1 c1(N2CCC(CNC(CCCC(C)C)=O)C23CC3)ncc2c(n1)CCCC2 N1(C(c2c(CC)ncs2)=O)CC(NC(c2ncc(C)cc2OC)=O)C(N=[N+]=[N-])C1 c1(CNC2C(C(=O)NCc3c(C)ccc(C)c3)C2)c(Br)ccc(Cl)c1Cl C1(C(=O)NCCCc2cc[nH]n2)C2CN(C(=O)C(C3CCOCC3)O)CC12 c1(C(=O)NC2C(C(N)=O)CCC2)cccc(Oc2ncc(Br)cn2)c1 C1(CNC(C(C(C)C)OC)=O)CCCC2CN(C(c3ccc(O)cc3F)=O)CC12 N1(C(CC2CCC(=O)N2)=O)CCN(C(=O)CCCF)CC1C(F)F CC(C)(C)CC(O)C(=O)N1CC(C2(Cc3cn(CC(F)(F)C(F)F)nn3)CC2)C1 C1(NC(Cc2nc(C(C)OC)sc2)=O)CC(O)CN(C(=O)CN2CC3CC3C2)C1 C1(CCC)CN(C(=O)CCCc2ccccn2)CCN1C(C1CC(C(F)F)C1)=O N1(C(C(=O)Nc2c(C)nccn2)=O)CCC2(O)CCCCC2(O)C1 c1(NC(C2C3CN(C(c4cccc(O)c4O)=O)CC23)=O)cccc(Cl)c1Br N1(C(C(CC)N(C(=O)CSCC(N)=O)C)=O)CC(F)(F)C(F)(F)C1 c1(CC)nc(=N)[nH]c(=NC(CNC(=O)Cc2ccc([N+](=O)[O-])cc2)C(C)C)[nH]1 CCCC(CCC)CC(=O)NCCCC1CCN(C(C2CCCCC2F)=O)CC1 c1(C(N(CCNC(COCCC#C)=O)CCOC)=O)c(C)cc(O)nc1C C(=O)(C(F)(F)C(O)C1CC1)N1CCN(C(CNC(c2cn(C)nc2Cl)=O)=O)CC1 c1(CC)oc(C)cc1C(N1CCCC1CN(C(=O)CC(=C)C)C)=O c1(C(=O)NCCC2(CNC(C3CC(C)C3)=O)CC2)ccc(Cl)c(OC(F)(F)F)c1 N1(C(C=CSC)=O)CC2CCC1CN2C(=O)C(C1CC1)C1CC1 C(C(C(=O)NCC(C)CNC(C1(C(N)=O)CCC1)=O)C(F)(F)F)OC N1(C(C(C)N(CC)CC)=O)CCCC(CC(=O)NCCn2ccccc2=O)CC1 c1(COC)c(C(=O)NCCC(=O)OC)cnn1-c1cccc(C)c1 N1(C(C(CC#C)(C)C)=O)Cc2ccc(CNC(c3cncc(Cl)c3C)=O)cc2C1 C1(NC(C2C(C(=O)OC)C2)=O)CC2CC(NC(=O)C(C)(C)n3cccn3)C1C2 C(CNC(=O)C=CC(C)C)(C(=O)NOCC1CC2C=CC1C2)OC N1(C(C(CC)O)=O)CC(N(C(=O)CNC(=O)Cn2cncn2)C)C2(CC2)C1 C(=O)(C(=O)C(C)(C)C)NC1CN(C2CN(C(CS(CC)=O)=O)C2)C(=O)C1 N1(C(C2=C(C)CCC2)=O)CC2CC(C(N3CC4CC3CO4)=O)CC2C1 Cc1cc(C(N2CC(N(C(=O)CCn3cccnc3=O)C)C(F)C2)=O)cc(Cl)c1 C12(C(=O)OC)CCC(C(=O)Nc3cc(CSC4(C)CCC4)c(F)cn3)(CC1)CC2 c1(C(N2CC3C(NC(C(C)NC(CC)(C)C)=O)C3C2)=O)cc(C)cc(Cl)c1 CC1CN(C(C2CC2(Cl)Cl)=O)CCC12CCOC2 C(CCCC(=O)N1CC(Cc2ccncc2CC(F)(F)F)C1)c1cn(CN)nn1 Cc1ccc(C(=O)NCC23CCCC2CN(C(C2(CO)CC2)=O)C3)c2c1CCC2 C1(C)(CC(=O)N(CC(=O)N(C)Cc2cnns2)C2CCC2)CCOC1 c1(-c2c(OCCC)nccc2)cnc2c(C(=O)NCC3CCC(F)C3)cccn12 c1(COC)nc(NCC2CN(C(=O)C(C)(C(C)C)OC)CCC2C)cc(O)n1 CC1(C)CCCCC1CC(=O)NCC=CCNC(c1ccc(=N)[nH]c1Cl)=O.C1CC1 c1(CN2CCCC3(NC(C(CC)CC(C)C)=O)C(C2)C3)cnc2ccccc2c1 N1(C(C(C(C)C)N(C)C)=O)CC(CNC(=O)C=Cc2ccco2)C2(CC2)C1 C1(NC(C2C(c3n(C)nnc3)C2)=O)CCCC(NC(C2CC(OC3CC3)C2)=O)C1 C12(C(=O)OC)CCCC1N(CC(=O)NC(c1cc(C)c(Cl)s1)=O)CC2 c1(C(N2C(CNC(C3(C)CCC(C)C3)=O)CC3(CC3)C2)=O)cnn2c1NCCC2 C(=O)(C#CC1CCCCC1)N1C(C)(CNC(c2c(C)nn(C)c2C)=O)CCC1 N1(C(C(CCOC)C)=O)CCOC2CCN(C(C3CN(S(N)(=O)=O)C3)=O)CC12 C(=O)(C1OCCn2ccnc21)N1CCC(CNC(c2ccn(C)c(=O)c2O)=O)C1 c1(N2CCC(CC=C)(NC(=O)Cc3cscn3)C2)nc2ccc([N+](=O)[O-])cc2s1 S(=O)(=O)(c1ccc(NC2COCC2N2CCCC2)nc1)N1CC(C)(C)C(CO)C1 C(=O)(CC(C)CC(=O)NC(C(=O)NOC1CCC1)C1(O)CCC1)OC O=C1NCc2c(C(=O)NC34CCCC3N(c3ncc(Br)cn3)CC4)cccc21 Cc1nnc(CNC(C2(O)CN(C(c3csc(Cl)n3)=O)C2)=O)n1C c1(C(=O)NCC(=O)NCC2C(CNC(C(C)C3CCCC3)=O)C2)ccccc1 c1(C(=O)NCC2CCC(C)(C)CN2C(=O)C2=CCC2)cc(S(N)(=O)=O)ccc1F O=C1C2CC3C1C3C2C(N1CCN(CC(=O)NCC(Cl)Cl)CC1)=O CCCC(O)CC(=O)NC(C)(CNC(c1ccc(OC)nc1)=O)Cn1cccn1 c1(C(N(C2CCN(C(c3ccc[nH]3)=O)C2)CC)=O)cnn(C)c1N C1(NC(c2cc(C)[nH]n2)=O)CCCCCCC1NC(C1CCC2CC12)=O N1(C(c2ccoc2Cl)=O)CCC(C2CCN(C(C3C4CC4C4CC34)=O)CC2)CC1 c1(C(N2CCOCC(NC(C3C(C)OCCC3)=O)C2)=O)scc2c1OCCO2 C1(NC(CCC#C)=O)CCC2(CCCN2C(c2cccc(SCC#N)c2)=O)CC1 c1(C2C(=C)C2C(=O)N(C)CCOCCNC(=O)CN(S(C)(=O)=O)C)ccccc1 N1(C(C(CC)OC)=O)CCCC1(C)CNC(c1cccc(C(F)(F)F)c1)=O C1(C(N2CCC(CNC(C3CC(C)OC3)=O)CC2)=O)C(C)(C)OC1(C)C CCC1=C(C(=O)NCC(C2CCC2)NC(C2CCc3nnnn3C2)=O)SCCO1 C(c1ccsc1Br)=CC(=O)NC1(CN(C(c2ccc(CC)[nH]2)=O)C)CC1 c1(C(N2CCCC(N(C)C(c3ccn(C(F)F)n3)=O)C2)=O)cc2ccncc2s1 n1(CCC(=O)NCCn2cnc(C(=O)NC(C3CC3)C3CC3)c2)cccnc1=O C(=O)(C(F)C(C)C(F)(F)F)NCC(CNC(c1cn(CCCC)nn1)=O)O CON(CCC(=O)NC)C(=O)CCSc1ccccn1 C1(c2ccccc2)(CNC(=O)OC(C)(C)C)CCN(C(C2C=CCCC2)=O)C1 c1(C(N2CCC(N(CCC)C(c3ncccc3F)=O)C2)=O)coc2ccccc12 c1(CN(C(=O)C(C)(C)c2ccsc2)C)ccccc1CNC(C1CNC(=O)N1)=O C1(C)(CNC(CC(C)(C)c2ccccc2)=O)CN(C(C2(C)CCCO2)=O)CCO1 S(=O)(=O)(c1ccc(Br)c(Cl)c1Cl)N(C(c1ccccc1N)C)C Cc1cncc(C)c1C(N1CCC(C(=O)N(C2COC(C)(C)C2)C)C1)=O C1(C(N2CCC(N(CC#C)C(c3coc(C(N)=O)c3)=O)C2)=O)COC(C)(C)CO1 C1(NC(C2CCCC(C)O2)=O)CN(C(=O)C(=O)NC2CC2)CC1S(C)(=O)=O CC1CC(CNC(=O)CCN(c2cnccn2)C)CCN1C(C1CC2CC2C1)=O C1(NC(c2ccc(OC)cc2Cl)=O)CN(C(C2CC3CCC2O3)=O)CC1C1CC1 c1(C(=O)NC(CCC#C)C(=O)N2CCOCC2)cc2cccn2cn1 C#Cc1cnn(CC(=O)N(CCCNC(=O)CNC(=O)CC(F)(F)F)C)c1 c1(C(N2CC(C)(CNC(C3(CC)CC3)=O)C(C)C2)=O)nccc2occc12 n1(CCNC(N(CC(=C)C)C)=O)ccc(C2CC2)n1 C1(C(N(CCO)CC)=O)CCCC(NC(c2cncn2C)=O)CC1 C(=O)(C#Cc1ccc(Cl)cc1)N1CCC2(C(C(N(C)C3CC3)=O)CCC2)C1 c1(C(N)=O)ccc(C(=O)NCC2CC2NC(=O)CCF)nc1 C#Cc1cncc(C(C(=O)NCC2CCOC(C)C2)N(CCCCCCC)C)c1 Cn1ncc2ncnc(N3CCC4CN(C(=O)C=Cc5cnccn5)CCC34)c12 C1(CNC(C(C)CCO)=O)COCCN(C(C2CCOC2)=O)C1 N1(C(C(N2CCCCC2=O)C)=O)CC2CS(=O)(=O)CC2(CNC(C2COC2)=O)C1 C1(NS(CC=C)(=O)=O)CCC(C(=O)NCc2ccc(O)nc2)OC1 N1(C(C2N(C(CCC(=O)OC)=O)CCC2O)=O)Cc2cccc(Br)c2C1 C(CCCCCc1nc(-c2nccs2)nn1C1CCCC(C)C1)SC N1(C(C2CCC(CNC(C3CC(N(C)C)C3)=O)O2)=O)CCc2nocc2C1 C1(NC(C(C(C)C)SCC)=O)CN(C(c2conc2C)=O)C2(CCCCCC2)C1 c1(CC)cc(C(=O)NCCC2CCC(NC(c3ccsc3C)=O)C2)sc1C C1(C(N2CC3C(CNC(CCSCC(N)=O)=O)(CC3)C2)=O)Cc2ccccc2O1 c1(C(N2CC(C3N(C(CC(CC)C)=O)CCC3)(O)C2)=O)ccc(OC)c(C)c1 c1(C(=O)NC(C)CC2CCCO2)n[nH]c2c1CN(C(=O)C(CN(C)C)N(C)C)C2 N1(C(C(=O)NCc2cccc(F)c2I)=O)CCC2(O)CCOCC2C1 N1(C(C2(CC)COC2)=O)CC2CCC1CN2C(c1c(Cl)cncc1Cl)=O Cc1nc(O)c(C(=O)NC2CN(C(C3CCS(=O)(=O)C(C)C3)=O)C2)nc1C N#Cc1cc(Cl)c(C(N2CC3CC3C2CNC(c2cccc(C(N)=O)c2)=O)=O)s1 C1(C(N2CCOC(CCO)C2)=O)(CNC(=O)C=CCF)CC12CCC2 c1(-n2c(C3(C)C(C)CN3)nnn2)ccc2c(c1)OCO2.C(C(C)(C)F)SC C1(C(=O)NC2(CNC(C(C)OC)=O)CCCCC2)CC(C)(C)OC1=O Cc1cc2c[nH]nc2cc1C(N1CCN(C(=O)C=CCO)C(CO)C1)=O c1(NC(N2CC(CC3CCCC3CF)C2)=O)cccc(F)c1 C1(C(=O)NCC2(NC(C(C)NC(CC)=O)=O)CCC2)Cc2nnc(C)n2C1 c1(C(N(CCN(C(CCC=C)=O)CCC)CC)=O)ccc(Br)cc1OC C1(C)(C(=O)NC2C(NC(c3scc(OC)c3)=O)COCC2)CCC(F)(F)CC1 C=CCC(C)(C)CC(=O)NC(COC(C)C)C(=O)Nc1csnc1C c1(C(=O)NCc2nc(CNC(Cc3ncc(C)o3)=O)sc2)ccc(Cl)c(F)c1F C(C)(CNC(c1ccn(C)c1C)=O)(CC(C)C)NC(CC(n1ccc(C)n1)C)=O C1(C(N(C2CCCC2)CCNC(C2CC(=C3CC3)C2)=O)=O)CC(F)(CO)C1 N1(C(C2(OC)CC(C)C2)=O)CCC(O)(CCNC(C2(F)CCCN(C)C2)=O)CC1 CCCCCCC(C)(C)C(=O)NCc1csc(CNC(=O)C2=CCOC2)n1 c1(OC)ncc(F)c(=NC(=O)c2cc(NC(C3(Br)CC3)=O)cn2C)[nH]1 N1(CC)CCN(C(C2(OC)CCN(C(=O)CN3CCC(F)CC3)C2)=O)CC1 C1(NC(=O)CC2(C(F)(F)F)CC2)CCC2CN(c3nc4ccccc4o3)CC2C1 C1(NC(=O)CC2C=CCC2)CCN(C(c2ncc(Cl)s2)=O)C12CCC2 C12(C(N3CCCC(NC(=O)CCC4OCCO4)C3)=O)CC1CCC2(F)F C1(C)(CC)CC(NC(c2cncs2)=O)CN1C(=O)CCc1cn(C)nc1C c1(C(=O)NCCC2CCN(C(C(C)=C3CC3)=O)CC2)cc(F)c(Cl)cc1Cl c1(C(=O)NC2(C)CC(NC(C3CCN4CCCC4C3)=O)C2)cc2ncccc2[nH]1 c1(CNc2cccc(OC(C)C#N)c2)c(Cl)cccc1C#N C1(OC)(CNC(=O)C(=O)N(C)C)CN(C(C2CCNC2=O)=O)C1 Cc1cn2cc(C(=O)NCC(C(C)(C)C)NC(c3cc(N)cc(F)c3)=O)sc2n1 c1(C(N2CCC(NC(Cc3n(C)cnc3)=O)CC2)=O)c(F)cccc1F N1(C(C(COC(C)C)NC(c2c(CC)cno2)=O)=O)CCC2OCCC2C1 CCC(C)(C)C(=O)C(=O)N1CCC(c2cn(C3CCCNC3=O)nn2)CC1C c1(OC)cccc(CN(C)CC2(OC(C(C)SC)=O)CCSC2)c1 N1(C(CC)=O)CCN(C(C2C3CN(Cc4cnc(C)nc4)CC23)=O)CC1 C1(CNC(C(C(C)C)NC(C)=O)=O)CCN(CC2C3CN(C4COC4)CC23)C(C)C1 CCCC(C(O)C(=O)NCC(C)(O)CC)NC(C12CCC(CC1=O)C2)=O c1(CC)cc(C(N2CC3CC3(CNC(=O)Cn3cc(CO)nn3)C2)=O)ccc1Cl C1(N(C(C(C)SCC)=O)C)CN(C(c2cc(Br)sn2)=O)CC12CC2 c1(NC(C(C)NC2(C(=O)OC)CCCC2)=O)cc(C(F)(F)F)ccc1[N+](=O)[O-] C1(CC(=O)N(C(C)CNC(=O)CC(C)(C)C)CC)CC2(CCC2)CO1 CCN=C(NCC=CBr)NCC1(CO)CCOC1 C1(NC(C(CC)NC(c2nc(CC)sc2)=O)=O)CC=C(C)CC1 c1(C(=O)NCC(C(C)C)NC(CN(C(=O)OC)C)=O)c(OC)ccc(Cl)c1F C1(CNC(CN(CC2(CC(C)=O)CC2)Cc2cccs2)=O)CCS(=O)(=O)C1(C)C C12(NC(CCNC(COC)=O)=O)CC(C(=O)NOCC3CCCC3)(C1)C2 C1(=O)CCC(C)(C)C(=O)O1.CC12CC(C(C(c3ccccc3)OC)=O)(CCO1)C2 N1(C(C(C)(C)CCCO)=O)C2CCCC1CC(NC(=O)COCC(F)(F)F)C2 C1(C(N2CCC(CSC)C2)=O)CC(=O)CN1C(C1CC(CC2CC2)C1)=O c1(C(=O)NCC2C(C)CCN(C(C(CC)=CC)=O)C2)cc2c(C)sc(C)c2s1 C1(OC)CC(CSC)N(C(c2ccc(C3CCCOC3)cc2)=O)C1 N1(C(C2(NC(C)=O)CCCC2)=O)CCC(CNC(c2cnc(C)s2)=O)C(C)C1 Cc1nc(Br)oc1C(=O)NC1CC(NC(=O)CCC(=O)c2ccc[nH]2)C1 N1(C(c2cnc(OC)nc2)=O)CC(NC(c2cc(N)ccn2)=O)C2CCCC2C1 N1(C(C(C)NC=O)=O)CCc2ccc(NC(C3CNCCO3)=O)cc2C1 CCC(C)C(CNC(C1(N(C(C2CCC(OC)C2)=O)C2CC2)CCC1)=O)CO c1(C(N2CCN(Cc3csc(Br)c3)CC2)C(=O)NCCC#N)cccc(Cl)c1 N1(C(CC)=O)CCOC(CCNC(c2ccc(C#N)s2)=O)C1 C1(NC(c2cnsc2)=O)CCC(CNC(=O)C(O)CN2CCOCC2)C1 N1(C(C(C2SC(=N)NC2=O)C)=O)CC(CNC(=O)CCC(C)(F)F)C(C)(C)C1 C(=O)(C(C)(O)CC(F)F)NCC(=O)NCC(c1ccc(OC)cc1)NC(C)=O Cc1cc(OCCC(=O)NCC(C)NC(=O)CCCN=[N+]=[N-])cc(C)c1 c1(C(=O)NC2CC(C)(NC(c3sc(CC)c(C)c3)=O)C2)ccc(N)c(C)c1F N1(C(c2ccc(COC)o2)=O)CCC(F)(C(=O)N(c2cccc(F)c2)C)C1 c1(C(=O)NCC(C2CCCC2)NC(c2ccc[nH]2)=O)cccc2c1OCCC2 C1(C(=O)NC2CC(OCC(=O)N(C3CCCO3)CC)C2)CC(=O)CS1 c1(CC)ccc(N)c(C(=O)NC(CO)C(C)NC(=O)CCn2ccnn2)c1 CCC(C)(C)C(O)C(=O)NC1CCN(C(c2cc(Cl)nnc2O)=O)C1C(C)(C)C C1(C(=O)NCC(=O)N(C)CC)CN(C(=O)C(C)(C2CC2)SC)CC12CC2 N1(C(c2scc(CC)c2)=O)CC(OC)CC1(C)CNC(=O)CN(C(=O)C(C)C)C CC(CCCCCO)N=c1[nH]c(=NC(C)c2ccc(Br)cn2)c2ncccc2[nH]1 c1(CN(C(C(CC)=O)=O)C(=O)OC(C)(C)C)c(C)cc(C)nc1C N1(C(CSc2c(OC)cccc2)=O)CCC2CC2(NC(=O)Cc2cc[nH]n2)CC1 c1(C(C(=O)NC(CCN(C(CCc2cc(C)no2)=O)C)C)C)ccc(F)cc1F CCC(C)C(CC(=O)NCC1(OC)CC1)NC(C1CCS(=O)CC1)=O C1(NC(c2c(CC)con2)=O)CCC2(CCCN(C(=O)Cc3csc(C)n3)C2)C1 N1(C(C2CC(C)N(C)CC2)=O)CCCC2(CC(O)C2)C1 N1(C(c2c(N)sc(C)c2C)=O)CC2(CCCC(CNC(C3CCC3(C)C)=O)O2)C1 c1(NC(C2CCc3[nH]nc(O)c3C2)=O)ncc([N+](=O)[O-])cc1NCCO C1(C(=O)NCC(C)(CO)NC(c2cc(C)c(O)nc2)=O)CCn2ccnc2C1 C1(CNC(c2ccn(CC(F)(F)F)n2)=O)CCCN1C(c1ccn(C2CC2)n1)=O c1(OC)cnc(F)cc1C(=O)NCC(C)(CO)NC(=O)CC1CN(C)CC1O CC1CC(C(N2CCCN(C(C3(c4ccn(C)n4)CC3)=O)CC2)=O)CCS1(=O)=O Cc1cc(O)nc(C)c1C(N1CC2C(NC(=O)CNS(=O)(=O)C(F)(F)F)C2C1)=O C1(C(=O)NCCCN(C2CCCC2)C(C2C(C(C)C)C2)=O)CCS(=O)(=O)N1 c1(CC)ncsc1C(=O)NCC1COCC1NC(=O)C(C)n1ccnc1 N1(C(C(CC=C)(C)C)=O)CCC(C2CC(NC(c3cc(OC)ns3)=O)C2)C1 c1(C(C(c2c(C)nc(C)s2)=O)C#N)cc(O)nc(=N)[nH]1 Cc1cnn(C(C)C)c1C(=O)NC1CC(NC(C2COC(C)C2)=O)C(O)C1 c1(C(C)OC)nc(C)c(C(=O)NC2COCC2NC(c2cnccc2Cl)=O)s1 C(=O)(C1=CCC(C)CC1)NC1CCN(C(c2ncc(CC)s2)=O)CC1C n1(C(C)C)ncc(C(=O)NCC23CC(NC(c4ccn(C)n4)=O)(C2)C3)c1N CCCC1c2ccccc2CCN1c1nc(C2CCCCC2)ns1 CCCC(C(=O)NC1CCN(C(=O)C(c2cnn(C)c2C(F)(F)F)C)CC1)OC C1(C(C)NC(CCCc2nc(C)sc2)=O)CCCCN1C(=O)Cc1cccn1C c1(OCCCC(=O)NC2C(NC(CC)=O)C2)cc(C(=O)OC)cc(Cl)c1OC c1(CN(C(C(=O)NCC(=C)C)C2CCSC2)C)ccc(C(C)(F)F)cc1 CC(O)(CC(=O)N1CCCC(O)(CNC(=O)CCc2ccncc2)C1)C(F)(F)F c1(C(N(CCCNC(c2nc(C(C)OCC)sc2)=O)C)=O)cc2ncccn2n1 c1(C(=O)NC2CCCC2NCc2c(F)cccc2Cl)cc(Cl)cc(Cl)c1[N+](=O)[O-] c1(OC)ccccc1-c1cc(C(N2CC3C(N(C(=O)C(F)OC)C)C3C2)=O)n[nH]1 N1(C(C2=CC(C)(C)C2)=O)CCCC2CCN(C(=O)COC(F)F)CC12 C1(NC(C2C(C)CCS2)=O)CCC(NC(c2cnn(C3CCCC3)c2)=O)CC1 Cc1cc(F)cc(C(=O)NCC(C)(O)CNC(c2cc3cccnc3s2)=O)c1C C12(CNC3CC4CCN(C(c5cc(CC)on5)=O)CC43)CC3CC(CC(C3)C1)C2 c1(C(N2CCC(O)(CNC(c3cc[nH]c3)=O)C2)=O)c[nH]c2cccc(Br)c12 C1(CC(=O)N(CC(=O)OCC)CC(C)C)CCCC(N)C1 C12(C(=O)NCC3(O)CC(C(=O)NC4(C(=O)OC)CCC4)C3)CCC(OC)C1C2 CC1CC(C)(C)CN1C(C1CC(NC(=O)CCN(C)CCO)C1(C)C)=O N1(c2ccc(C(=O)OCC)cn2)CCC(C)C(NC(c2ccon2)=O)C1 C(C(C)(C)CC(=O)N1CCCC(C(=O)NCCN2CC=C(C)CC2)CC1)OC C1(NC(=O)CCCc2cc[nH]n2)CC2CCC1CN2C(=O)CC1(CO)CC1 C=CC(C)(CCOC)C(=O)NC1CC2CN(C(c3ccc(O)nc3)=O)CC2C1 N1(C(C(CCOC)C)=O)CCCCCC(NC(c2cc(C(F)(F)F)ns2)=O)C1 OC1CCC2(CC1)CCN(N1CCOC(c3ccccc3)C1)CC2 Cc1ccc(C(C)C(=O)NCCOCCNC(C2CN(C(N)=O)C2)=O)s1 N1(C(C(C)n2cccc2)=O)CCCC(CNC(c2cc(F)n(C)n2)=O)C1 c1(COC)ccc(C(=O)NCC(O)CN(C)C(c2cc(C)sc2C)=O)cc1F N1(CCNC(c2ccsn2)=O)CCN(C(c2ccn(C(C)(C)C)c2)=O)CC12CCC2 C1(NC(=O)C(c2cccc(Cl)c2)O)C2CCC1CN(C(=O)Cc1ccccc1)C2 C1(NC(c2cncc(C)c2)=O)CC2CC1CN(C(C13CCC(C)(C1)OC3)=O)C2 C1(C(=O)NCCCOCCC(=O)N(CC#C)C)CC2C=CC1C2 N1(c2c(C)c(Cl)ncn2)CCC2(CC1)CC(NC(C1CCS(=O)(=O)C1)=O)CCO2 C(C(F)(C(=O)NC(C12CCC(CC1)C2)C)C(C)C)NC(c1cccc(OC)n1)=O C(=O)(C1CCc2ccccc21)NC1(C)CC(NC(c2cc(C(N)=O)[nH]n2)=O)C1 c1(OC)ccc(CNC(=O)C(O)CNC(=O)C(F)OC(F)(F)F)cn1 Cc1cc(C(N2CC(CNC(=O)C(C)(C)C3CC3)C3CC23)=O)c(Cl)cc1F c1(C(=O)NCCC(C)NC(=O)C(c2ccc(Cl)cc2)O)ccc2nsnc2c1 CCC(Cc1nc(CCSC)nn1-c1cccc(C(C)C)c1)C(F)F N1(C(c2ccc(CCC)cc2)=O)CC(OC)C(OC)C1CNC(c1cn[nH]c1)=O C#CC1CCN(C(=O)CC2CC(O)CN2C(=O)Cc2cccs2)C1 c1(C(N2CC(CCNC(C3CCC4(CC4)C3)=O)OCC2)=O)ccc([N+](=O)[O-])cn1 N1(C(c2c(OCC)scc2)=O)CCc2sc(CNC(=O)C(C)(C)C#N)nc2C1 N1(CC(c2cncc(C)c2)=O)CCC(CO)C(c2ccccc2)C1 C=CCC(C)(C)C(=O)NCC(C)(C)CNC(=O)C=C(C)c1ccsc1 C(=O)(C(O)CC(C)(C)C)N(CCC)CCNC(C1(C2CCCO2)CC1)=O O=[N+]([O-])c1cc(F)ccc1CNC(=NCCCF)NCC1CC12CCSCC2 c1(SCC(=O)NC2CN(C(=O)CO)CC(C)(C)C2)ccc2c3c(cccc13)CC2 c1(CNC(C2CCCN2C(c2cnc(Cl)cc2Br)=O)=O)cccc2cnccc12 CC(CC(=O)NCc1conc1C1CC1)C(C)(C)NC(=O)CCCCN=[N+]=[N-] c1(C(c2csc(CN3CCCC(O)C3)n2)C)nc(-c2cc(Cl)ccn2)nn1CC C(=O)(CCCCCC#N)N1CCC(CCCCNC(C(CC2CC2)OC)=O)CC1 C(=O)(C(C)C(F)(F)C(F)F)N1CCC(CNC(C(CC=CC)C)=O)CC1 c1(C(=O)NCC2CCN(C(C(C)=C3CC3)=O)CC2)ccc(C)c2cccnc12 N1(C(C(C)Cn2cccn2)=O)CCCC1(C)CNC(c1cc(C(F)F)nn1C)=O c1(CC)cccc(N(C)C(=O)NCC2CCCOC2c2nccn2C)c1 Cc1cc(N)c(C(=O)NC(C2CCN(C(=O)C(C)C3CCOC3)C2)C)c(F)c1 c1(C(=O)NCCC2(O)CN(C(Cc3c(C)nc[nH]3)=O)C2)cccc(O)c1Cl c1(C(=O)NC(C(=O)NCCC(CC)(F)F)C(C)CC)ccn2cncc2c1 c1(OC)cccc(C(CC(=O)O)NC(C2CC2c2cnn(C)c2)=O)c1 N1(C(c2ccnn(C)c2=O)=O)CCC2(CC1)CN(C(=O)CCCc1cncs1)C2 c1(C(N(C)CC2CCN(C(c3cc([N+](=O)[O-])n[nH]3)=O)C2)=O)cnn2cnnc2c1 C1(CC(N)=O)CN(C(c2cnc(C3CCOC3)s2)=O)CCN1C(c1cnn[nH]1)=O C1(CC(=O)NCC(C(C)C)NC(c2ncncc2F)=O)(COC)CCOCC1 N1(C(COCCOC)=O)CC2CC2(C(=O)Nc2cc(OC)ccn2)C1 c1(OCC(=O)N(C(C2CCCO2)C)C)ccccc1CNC N1(C(C2(C)C(C)(C)C2(C)C)=O)CCC(NC(=O)Cn2nnc(=O)[nH]2)C(F)(F)CC1 CN=c1[nH]c(=NCC2CCC2(F)F)[nH]c(=NCCN2CCS(=O)(=O)CC2)[nH]1 C1(CNC(COCCC#C)=O)CN(C(=O)CCOCCOC)CC(C)O1 C(=O)(CCCCN(C)C)NCCN(C)C(c1ncccc1OC(F)F)=O n12cc(nn1)C(=O)NCC2.C1(NC)CC(CC(=O)NCCCc2nncs2)C1 c1(OCCC)cccc(CC(N2CCC3C(NC(=O)CSCC(C)C)C23)=O)c1 C1(NC(C2CCCO2)=O)CN(C(=O)CCOc2ccccc2)C2(CCC2)C1 c1(NC(=O)C(N2CCOC(CC3CCCC3)C2)=O)cccc(CO)n1 N1(C(=O)C2=CS(=O)CCC2)CC(C2CCCN(C(c3cnoc3C3CC3)=O)C2)C1 CC1CSCCN1C(C1(CNC(=O)C=Cc2ccoc2)CC(C)(C)C1)=O C1(C(=O)NC2C(=O)NCC2)C2CC2CN1C(=O)CCC1CCCCO1 N1(C(C(C)NS(C)(=O)=O)=O)CC2CC(NC(c3cc(Cl)c(Cl)n3C)=O)C1C2 C=CC1CC(N=c2[nH]c(=NCCc3cccc(C)c3C)[nH]c3cc[nH]c23)CCO1 CCCS(=O)(=O)CC(=O)NC1CCC(C)N(C(C2CC2(Cl)Cl)=O)C1 N1(C(=O)NCc2nc(OCC)sn2)CCN(C(=O)CN(CC)CC)C2CCCCC12 c1(C(C)C)ccc(F)cc1C(=O)NCC1CC(F)(CNC(=O)CS(N)(=O)=O)C1 c1(CCC(=O)NC2C(NC(C3CCN(C)C3)=O)CCC2)cc2ccccc2o1 c1(C(=O)NC2C(NC(C(C)CC3CC3)=O)C2)ccnc(NCCN(C)C)c1 C1(CC)CCN(C(=O)CN(C2CS(=O)(=O)C2)C)C1NC(c1cn(C(C)C)cn1)=O N1(C(C2CC(NC(C(C)CN(C)C)=O)C2)=O)CCCCC1Cc1ccccc1 CCCCC(CC)CC(=O)NC1CCN(C(c2nc3c(s2)COCC3)=O)C12CC2 N1(C(C#CC(C)(C)C)=O)CCC2(CC1)CN(C(C1CCn3ccnc3C1)=O)C2 C(=O)(C1CCc2c[nH]nc21)N1CCC(OC(C(=O)OCC)(CC)CC)CC1 N1(C(C2=C(C#N)CCC2)=O)C2CCC1C1CC1(NC(C13CCCN1CCC3)=O)C2 n1(CC)nc(C(N2C(C(=O)Nc3cccc(COC)c3)CC2C)=O)cc1C c1(CC(C)NC(C(F)=CC)=O)ccc(CNC(C2CCOC2)=O)cc1 C1(C(=O)NC(c2ccc(F)cc2)CCC)CSCCN1C(c1ccnc(C)c1)=O c1(C(=O)NCC(C)C)ccc(-c2cccc(CC(N3CC4(CCC4)C3)=O)n2)cc1 C1(CC(N2CC(CC(C)NC(=O)CN3C(=O)CNC3=O)C2)=O)CC(F)(F)C1(F)F C(=O)(C(C)(C)CC(=O)N(C)CCC1CCN(C(C23CC(C)C2C3)=O)CC1)OCC c1(C(N2C(C(C)NC(=O)Cc3ccco3)CCC2)=O)cccc(C#N)c1 C(=O)(CCCc1cc(C)no1)N(C1CCCC1)CCNC(CC=C)=O c1(N2CC(=O)OCC2)ccc(C(C)CCO)cc1.c1(OCC)ccccc1.C(C)(C)(C)O C1(O)(CNC(C(CC)CC2CCCC2)=O)CCCN(C(c2cnc(OC)s2)=O)C1 c1(CC(C(=O)NCC2CCCN(C)C2)NC(C(CC)OC)=O)ccccc1Br C#CCC(C)(C(=O)N1CCC(CC)CC1)NC(c1cc(=N)[nH][nH]1)=O N1(C(C2(CC#C)CCC2)=O)CCC(NC(c2ncc(C)cc2F)=O)C(CC)C1 C1(NC(c2n(CC)cnn2)=O)C(C)CCN(C(=O)CC2CCNC2=O)C1C N1(c2c(OC)cnc(SC)n2)CCC2C1CCCN2C(c1cc(Cl)c(Cl)cn1)=O c1(C(=O)NC(c2ccncc2)CC)c(NCc2cnc(OC)nc2)cccc1F N1(C(C(N2C(C(=O)OC)CC3(CCC3)C2)=O)=O)CCc2ccc(C)cc21 n1(CC(=O)NC2CC(F)(CNC(C3CSC3)=O)C2)cnnc1O C1(CNC(C2CC3CCC2CC3)=O)CC(F)(F)CN1C(c1cn(C2CC2)cn1)=O N1(C(C(C(=C)C)(C)C)=O)CCC2CCC(NC(=O)COC3CCC(C)CC3)C1C2 CC(C)CC(C)CC(=O)NC1CC(C)(NC(=O)C(C(C)O)N(C)C)C1 CCCC(C)C(=O)NC1CCC1CNC(c1cnn(CCOC)c1C)=O CC(C(=O)NCCC1CSCCN1C(=O)CNC(c1cccs1)=O)C1=CCCC1 C1(CC(=O)NC)CC2(CC2)CN1C(c1ccnc(OC)c1Br)=O N1(C(c2ccc(C)s2)=O)CC2CC2(C(=O)Nc2ccnc(C3CC3)c2)C1 C(=O)(CC1=CCN(C)CC1)NCCC1(OC)CN(C(=O)C(O)C(C)C)C1 C1(NC(C(C)c2cccs2)=O)CCN(C(=O)C(C)CN2CCOCC2)C1 c1(NC2(CC(C)C)CC2)nccc2cc(F)ccc12 Cc1cc(COCCOCCOCCOC(c2ncc(Cl)cc2Cl)=O)ccc1F N1(C(C(CC)(C)COC)=O)CC2(CCN(C(=O)CC3(O)COC(C)(C)C3)C2)C1 c1(C(=O)NC2CN(C(CC(C=C)CC)=O)C2)cc(OC)cc2cccnc12 N1(C(CC2N(CC)CCC2)=O)CCCC(c2cn(CC3CC3)nn2)CC1.O C1(C#N)(C(N(CCCCNC(C2CCC2c2nc[nH]n2)=O)C)=O)CC2CC2C1 N1(C(CCC(=O)NC)=O)CC2CC(C1)CN(C(=O)C(C)c1cncs1)C2 CC(C)C(C(=O)N(C)CCSc1ccccc1)CNC(=O)CC1CCC(C)CO1 c1(CC(=O)NC2C(CNC(C(COC)(C)C)=O)CCCC2)c(C)cccc1C C1(C(N2C(C(N(C3C=CC(CO)C3)C)=O)CCCC2)=O)CCC2CC1CO2 C1(NC(=O)C2CC2)COC2(CNC(C3CCCN3C(=O)C(F)(F)F)=O)CC1C2 N1(C(=O)CSCCN2CCCC2)CC2(C1)CN(C(c1ccccc1F)=O)CCO2 C12(CNC(=O)CC3OCCO3)CC1CN(C(c1cn(C(F)F)nc1C(F)F)=O)C2 N1(C(c2c(C)nco2)=O)CCN2CCN(C(C3CCCSC3C)=O)CC2C1 c1(OC)c(C(=O)NC2CC(CCNC(=O)C(C)Cc3ccncc3)C2)csc1Cl c1(CNC(c2nnnn2CCCOCC)C2(CCC)CC2)ccn2ncnc2c1 C(=O)(C(C(C)(C)O)NC(=O)CCNC(=O)OC)NC(C(CC)CC)C C1(C(=O)NCC2N(C(C3(C(=O)OC)CC3C)=O)CC2)CSCN1C C1(NC(CCN(CC(F)(F)F)C)=O)CN(C(C2(C)COC(=O)OC2)=O)CC1(C)C N1(C(=O)NCC2(C(C)(C)OC)CC2)CC(C)(C(=O)O)C(F)(F)C1 c1(C(N(CCCNC(C23CCC2C3)=O)C)=O)scc2c1CCCC2 c1(OC)cc(C(=O)NC2CC(NC(C3CCC(C)(C)C3)=O)C2)cc([N+](=O)[O-])c1N C1(c2nn(-c3cc(F)cc(F)c3)c(C3CC3C(F)F)n2)CCc2ccccc2C1 S(=O)(=O)(c1cccc(Cl)c1)NC1C(C)CN(C(=O)Cc2cccnc2)C1 c1(C(N2CCC(C(=O)NC34CCC(CC3F)C4)CC2)=O)ccc2nccn2c1 C(CCC(C(=O)N1CC(SCC(F)F)C1)NC(=O)C(C)S(N)(=O)=O)OC n1(-c2cc(C)on2)c(C)cc(C(=O)CN2CCC(c3nncn3C)CC2)c1C CCC(CC)CC(=O)NCC(C)C(=O)NCCC(=O)NC(C)C c1(C(=O)NCCC2CCN(C(C(F)=C(C)C)=O)C2)ccc2c(c1)CCCCC2=O CC1C(NC(C2CCC3(CC3)C2)=O)CCCN1C(c1nc(C2CC2)ncc1Cl)=O C12(C(N3C(C)CC(CNC(=O)Cn4cc(Br)cn4)C3)=O)CC(C)(CCO1)C2 Cc1ccc(C(=O)NC2C=CCCC2C(=O)N(CC(C)C#N)C)nn1 Cc1cc(C(N2CC(F)CC2CNC(C2CCCCC(=O)N2)=O)=O)cnc1C c1(CC(N2CC(O)(C(CNC(C(Br)=C(C)C)=O)(C)C)C2)=O)cccnc1C C1(CNC(C2C(C)C2C)=O)CC(F)(F)CN1C(=O)C(O)Cc1ccc(F)cc1 c1(C(=O)OCc2nnc(C)n2-c2ccccc2)cc(I)ccc1Br N(C(=NCC(C)C)NCC1CC12CC2(F)F)Cc1ncn(CC)c1 C1(C(N(CCCNC(C(C)N(C(C)=O)C)=O)CCO)=O)CCc2nccn2C1 CC1CCN(C(c2ccc(F)s2)=O)CCN1C(=O)Cc1ccc(Cl)c(F)c1 c1(C(=O)NC(C(C)(C)NC(C2CC(C#N)(OC)C2)=O)C)cc2n(c1)CCCC2 N1(C(C2(CO)CC(C)(C)C2)=O)CC2CN(C(=O)C(C)(C)F)CC2(C)C1 N1(C(C2C3CNC(=O)C32)=O)CCN(C(c2cnc(C3CC3)o2)=O)CC(O)C1 C1(C)(C(=O)NC(C)CC2CCCCC2)CC(O)CN1C(c1c[nH]nc1Cl)=O CC1(C)CN(C(c2cocn2)=O)CC1NC(C1CCN(C(=O)OC(C)(C)C)C1)=O C12(CNC(CC(CC)C)=O)CCC(CNC(C3C4CCCC34)=O)(CC1)OC2 C1(C(=O)OC)CCC(C(=O)NC2(CNC(=O)CCOC(C)C)CCC2)C1 C1(SCC)CCC2(CC2)N1C(=O)CC(C)(C)C1CC1 CCC(C(=O)NCC1CC2(C1)CN(C(c1c[nH]c(C(N)=O)c1)=O)C2)C(C)C O=C(C1CCc2nccn21)NC1C=CCN(C(=O)C=CCN2CCOCC2)C1 O=C(N=c1cc[nH][nH]1)NNC(=O)c1cc(F)cc(F)c1 C1(NC(C2(CCOC)CCCC2)=O)CN(C(c2nc(O)c(C)s2)=O)CCC1F CCCCC(O)C(C)C(=O)N1CCC(CCC(N2CC3OC(=O)N(C)C3C2)=O)C1 C12(CN(C3CCCCC3)C(C)C)CC(COC)(CO1)C2 CC1CC(N2CCCC2)CN1C(C1CNC(=O)O1)=O N1(C(CCC=C(C)C)=O)CC(CNC(c2c[nH]ccc2=N)=O)C(C)C1 N1(C(C)=O)CC2(NC(=O)C3=CCCCO3)CCC1C2 c1(C(N2CCC3(NC(C4CN(S(C)(=O)=O)C4)=O)C(C2)C3)=O)ccc(Cl)c(Cl)c1O C1(CNC(c2cncc(C3CC3)c2)=O)CCN(C(=O)CCC2CCCO2)CC1 C1(NC(Cc2cnc(OC)nc2)=O)C2CC3CN(C(=O)C=C(C)C)C1C3C2 c1(C(=O)NCC(C2CCCC2)NC(C(C(C)C)OCC)=O)cc(N)c(Cl)cn1 N1(C(C(CC(=C)C)OC)=O)CCC(C)(C)CC1C(N1CC(F)(F)CC1CO)=O C=CCCCCC(=O)NC1CCCCC1CNC(c1ccc(F)s1)=O CCCCC(CC)CC(=O)NC1C2CC1N(C(c1sccc1F)=O)C2C S(=O)(=O)(c1ccc(=NCC2OCCc3sccc32)[nH]c1)NC1CCC(C)(C)C1 Cn1nccc1C(=O)NC1CN(C(c2nscc2I)=O)C1 c1(C(=O)NCC(C)CNC(C2CC2c2cccnc2)=O)cc2c(s1)COCC2 C(N=c1nc(N2CCCC(CN(C)C)C2)c2c([nH]1)CCS2)c1cnc(C)s1 CC1CN(C(C(=O)NC2CCC2)c2nccs2)c2cc(Cl)ccc2O1 c1(C(c2nnnn2C(C)C(=O)OC)NCCOC(C)=O)nn(C(C)C)cc1Cl c1(CC(C)C)c[nH]c(C(=O)NCC2(O)CC(CNC(C3(O)COC3)=O)C2)c1 CC1CCC(Cl)=C(C(=O)N(C)CC2CCN(C(C3CC(F)(CO)C3)=O)CC2)C1 C1(NCC(=O)NCC(C)(C)NC(C2C(C(=O)OC)COC2)=O)CCC(F)(F)CC1 C(C(=O)N1CC(NC2C(CNC(c3ccc(CO)s3)=O)CC2)C1)(C(C)C)OCC CC1CC(NC(=O)C(F)(F)c2nccs2)CN(C(c2cc(N)c(F)cn2)=O)C1 N1(C(Cc2cn(C(C)C)nn2)=O)CCN(C(C2CCCC(F)(F)C2)=O)CC(C)C1 C(CCN(C(=O)C(CCOC)OC)C)(C(C)C)NC(C1(CCC=C)CC1)=O C(C1CCOc2ccccc21)NC(=O)Nc1ncc(C)nc1 C1(NCC(N2CC(F)CC2CNC(C23CC(F)(C2)C3)=O)=O)CCS(=O)(=O)C1 N#Cc1c[nH]c2ccc(C(N3CC(CC(=O)Nc4ccc(F)cc4O)C3)=O)cc12 N1(C(C2OCCC(=O)C2)=O)CC2(CCNC(c3csnn3)=O)CCC1CC2 C(CC(N=c1[nH]c(Cl)ncc1Cl)C(C)C)NC(C(C)SC)=O C(=O)(CCCCCNC(c1cc(C#N)cs1)=O)N1CC(CC(C)C)OCC1 C(CCCCNC(C1(C#N)CC1C(F)(F)F)=O)N(C(CCSCCCC)=O)C C1(NC(C(CC)OC2CCCC2)=O)CC2CC(C1)N(C(c1nnn(C)c1C)=O)C2 N1(C(CC(=O)OCC)=O)CCC(C(F)(F)F)C(NC(C2(CF)CC2)=O)C1 N1(C(Cc2c(OC)cccc2)=O)CC(N(C(=O)C(C)C(F)(F)F)C)C2(CC2)C1 C12(C(=O)NCC(CC)(C)COC)CC(CCO1)N(C(=O)CC1CC1(C)C)C2 c1(OCCC)ccc(Cl)cc1CC(=O)NC1CCN(C(=O)C2=CCCC2)C1C C(CCN=c1[nH]c(C2CCCC2)cs1)N(C(=O)OC)C c1(C(N2CC3C(C(=O)Nc4cncnc4Br)C3C2)=O)c(Cl)cccc1Br c1(C(=O)NCCC2N(C(c3ncc(OC)nc3)=O)CCCC2)cccc(N)c1F N1(C(C2CCC(C)C2)=O)C(CC(=O)NCC=Cc2ccccc2)C2CCCC12 c1(CCNC(=O)C(Cc2ccoc2)NC(C2COCCOC2)=O)nccc(O)n1 CC(C(=O)NCC(C)(C)C(=O)NCc1cccc(CO)n1)C(F)(F)F CN1CCCCC1C(N1CCCCC1C1(CNC(=O)CC(C)(F)F)CC1)=O N1(C(CC=CC=C)=O)CC2CC1CN2C(c1cccc(I)c1O)=O C(=O)(C(CC(C)C)NC(C1CC1CCC)=O)N1CCCC(OCC#C)C1 N1(C(Cn2cc[n+](C)c2)=O)CC(C)(CNC(=O)CC2CCCOC2)CC1(C)C N1(C(CCCN(C)C)=O)CCC2CC1CN(C(=O)CS(=O)C(F)(F)F)C2 N1(C(C(C)=C(C)C)=O)CCN(C(c2cccc3c2NCC3)=O)CC12CC2 C(C(=O)NC1CCN(C(=O)CCc2cccs2)CC1)(C(C)C)NC(C)=O C1(C(=O)NCCOC2CN(C(CC(CC)O)=O)C2)COc2ccc(OC)cc2C1 c1(C(=O)NC2CC(NC(CCCC(=O)NCC)=O)C2)sc2nccc(C)c2c1C c1(OC)cscc1C(N1CC(N(C(=O)CC2CCOC2=O)C)C1)=O C(=O)(C(C)CC(C)(F)F)N1CCN(C(CCC(=O)N(C(C)C)C)=O)CC1 c1(CC)nn(C)cc1CNC(=O)Nc1nccc(-n2nc(C)cc2C)n1 N1(C(C2CC(SC)C2)=O)CCOCC(NC(c2cccnc2C)=O)C1 N1(C(Cc2ccc(C#N)cc2)=O)CC2(CCCN2C(c2ncccc2F)=O)C1 O=S(=O)(c1ccc(NC2CCOCC2OC(F)F)nc1)NCc1ccnnc1 CC1(C)OC(=O)CC1C(=O)NC(CNC(c1csc(Br)n1)=O)CO c1(N(CC(N2CCCC(NCC=CC)C2)=O)CCC)ccc(C#N)cn1 C12(C(N3CCC(N(CC#C)C(C4CC(C)C4)=O)C3)=O)CCCN(CC1)C2 c1(C(=O)NCC(C2N(C(CCNC(C)=O)=O)CCCC2)C)cc(Cl)n[nH]c1=N c1(C(N2CCC(N(CCO)C(c3ccc(O)nc3)=O)C2)C)ccc(F)cc1 c12c[nH]c3ccc(cc13)[nH]c2=O.N1(Cc2c(C)noc2C)CCCC(O)C1C CC(C)CC(CC(=O)N(C1CCCCC1(C)C)C)NC(C1CCN(C)C1=O)=O C(=O)(C(C)C(=O)NC(CNC(=O)Cc1cncc(C)c1)C1CCC1)OC CC1CCN(C(=O)CCn2cc(-c3ccc(Cl)c(Br)c3)nn2)CC(C)O1 C1(C(=O)NCC23C(CN(C(C4(C)CC=CC4)=O)C2)C3)CC2CCC(C1)C2 c1(-c2nc(NC(=O)NCC3(CF)CCOCC3)sc2)ccc(Cl)cc1Cl CCCN=C(NCC(CC)Oc1cccc(F)c1)NCC1(F)CCOC1 C(=O)(C(CNC(=O)C(F)Cc1ccccc1)CC1CCCC1)NC1CCC(=O)C1 c1(C(=O)NCCC(C)NC(c2n[nH]cc2C2CC2)=O)ccc2c(c1)C(=O)NC2=O N1(C(C(C)c2ccsc2)=O)CCN(C(C2CCCCC2O)=O)C(C)C1 CC(C)CCN=C(NCC(N1CCN(C)CC1)C(C)C)N1CCCC(C)(F)C1 CC(CCNC(=O)NCc1cn(CC2(c3ccncc3)CC2)nn1)C(=O)O c1(C(=O)NCCN(C(=O)C=Cc2ccsc2)CC)cnc2n1C(C)CCC2 N1(C(CCC#C)=O)CC2CCC(NC(=O)Cc3cccc(F)c3OC)(C2)C1 C(=O)(C(CCC1CC=CCC1)N(C1CC1)C(c1cccnc1)C)NCCCCCC CC1CC(C(=O)NC2CCCC2CC(=O)NC(c2nncn2C)CO)CC(=O)N1 C(c1ccc(F)c(F)c1)=CC(=O)NC12CCC(C1)N(C(C1CC1CF)=O)C2 C=CC1CN(C(C(=O)NCc2cccc(Cl)c2)C(C)C2CCCOC2)CCO1 N1(C(CCCC(=O)NC(C23CC4CC2C3C4)=O)=O)CCN(C(C)=O)C2CCCC12 C(=O)(C(CNC(=O)CN1CC(C)(C)C1)CC1CCCC1)NC(COC)(C)CO c1(C(N2CC(NC(c3c(C)cccn3)=O)C(F)C2)=O)ccc2nonc2c1 C(=O)(C1=CCCCCC1)N1C(CC(=O)NCC2CCC3(CC3)C2)C2CCC1C2 S(=O)(=O)(c1cc(Cl)cc(Cl)c1)N1CC(NC(c2ccc(Cl)c(Cl)n2)=O)C(O)CC1 C(=O)(C(CNC(c1ccn(C)c(=O)c1)=O)(CC)CC)NC(C#C)C(C)OC CC1(c2cn(Cc3ccc(Br)s3)nn2)CN(C(c2csc(I)n2)=O)C1 C(C)(CO)(C(=O)NCC(C)CN(C(=O)CCCc1csc(C)n1)C)OC C1(OCCNC(C=CC(C)(C)C)=O)CCN(C(c2csc(S)n2)=O)C1 C1(CC(=O)NC2CCC(NC(c3nnn(C(C)(C)C)n3)=O)C2)C(=O)NN=C1C c1(C(=O)NCCN(C(=O)CCCCNC(=O)OC(C)(C)C)C)cc([N+](=O)[O-])n[nH]1 S(=O)(=O)(c1cc(C)cnc1NCC1OCCOC1(C)C)NC(CC)CCOC C(N(C)N1CC(O)(c2nnnn2CCCN2CCCC2)C1)C1CN(C)C1 N1(C(CC(C)(C)C(F)F)=O)CCc2ccccc2C(NC(C2CCC3CC23)=O)C1 O=S(=O)(c1ccc(NC2COc3cc(F)ccc32)c(F)c1)NCCCCCO N1(C(COCC(=O)NC)=O)CCC2CCCC12CNC(c1coc(SC)c1)=O C1(NC(C(C)Oc2cccnc2)=O)CCC(CNC(c2cc(C(N)=O)c[nH]2)=O)C1 CCC(C)(CCNC(=O)CC(C)(O)c1ccccc1)NC(=O)CSC(C)C N1(C(CCCC(=C)C)=O)CCC2CC(NC(C34CC=CC(C3)OC4)=O)CCC2C1 C1(CNC(c2cc(Cl)cs2)=O)CC(C(F)(F)F)CCN1C(C1CCCSC1)=O Cc1noc2nc(C(N3CC(NC(c4c[nH]nc4F)=O)C(O)C3)=O)ccc12 CC(CN(C(=O)CC1CN(C(C2CN3CCC2C3)=O)CCO1)C)C(F)(F)F CC(CC(F)F)C(=O)N(C1CN(C(c2c[nH]nc2-c2ccsc2)=O)CC1(C)C)C C(c1ccc(O)cc1)=CC(=O)Nc1scc(CNC(C(C)O)=O)n1 c1(CNC(C(C)CN(C)C)=O)cnn(C)c1C(N1CC(CCO)C1)=O N1(C(c2n(CC)ccc2)=O)CC(CNC(c2ccncc2)=O)C(C)(C)C1 C1(CC)CCCC(NC(C2(CNC(=O)CCN3CCCC3)CC(C)(C)C2)=O)C1 c1(C(N2CC(N(C(=O)CC(C)(C)C(F)F)C)C2)=O)ccc2cncnc2c1 N1(C(Cc2cc(C)on2)=O)CC2CC2C1C(=O)NC1COCCC1O c1(C(=O)NC2(COC)CCCN(C(=O)C(C)CSC)C2)cn2c(n1)CCCC2 N1(C(CNC(=O)NC)=O)CCN(C(c2cccc(-c3ccncc3)c2)=O)C(C)C1 CC1CCN(C(c2cnn(C)c2Cl)=O)CC1N(C)C(C1CC2(C1)CC21CC1)=O C1(CNC(COC2(C)CCCC2)=O)CC2CCC(C1)N2C(C1(C)CCNC1=O)=O C1(C)(CNC(CNC(C)=O)=O)CN(c2nc(C(C)C)ns2)CCO1 C1(CCNC(CN(C)CC)=O)CCCN(C(c2cnnc(C)c2)=O)C1 C(=O)(CCCC(F)F)N(CC)CC1CCC(C2CC2)O1.N12CCC(CC1)CC2=O c1(CC)cccc(NC(=O)C#CCNC(C2CCCC(C)C2)=O)c1F CON(C)C(=O)C1(NC(C2CCOCC2)=O)CC1 c1(C(=O)NC2CCN(C(C3(C=C)CCCCC3)=O)CC2)c(F)cc(C#N)cc1F C1(NC(CC(CCC)NC(C(CC=C)(C)O)=O)=O)CC12CCCCCC2 c1(-n2cc(CN3CCC(NC(c4scc(C)c4)=O)C3)nn2)c(C)noc1C N1(C(Cc2nnc(C)o2)=O)CCC(C)N(C(C2CC(=O)N(C3CC3)C2)=O)CC1 C#CC#CC(C)(C)NC(C1CCC(NC(=O)C(C2CCOCC2)F)CC1)=O C(=O)(C#CC1(C)CCCO1)N1CCC(NC(c2c(O)ccc(OC)c2)=O)C1 CCC(C)(C)C(O)C(=O)NCC1CCCN1C(c1cncc(F)c1)=O C1(CC(=O)NCC2CCC2)CN(C(=O)CCNC(C2CC(OC)C2)=O)CC1C n1(C2C(=C)C2)c(-c2cn(C)nc2C(=O)OCC)csc1=Nc1ccc(F)c(F)c1 c1(C(=O)NC2(C)CCN(C(C(CC=C)C)=O)C2)ccc2c(n1)CCCC2 O=S(=O)(Oc1cccc2c(I)cccc12)C1CC(C2CCC2)C1 N1(C(C(C)CC(N)=O)=O)CCCC12CCN(C(C1(C(F)(F)F)CCC1)=O)C2 c1(C(=O)NCC2OCCC(NC(C(CC)(C)C)=O)C2)cc(C#N)oc1C c1(NC2(c3n(C(CC)C)nnn3)CSC2)cc(C(=O)OC)cnc1OC N1(C(CCCC)=O)CCC2C(CCCN2C(C2CN(S(N)(=O)=O)C2)=O)C1 c1(C(c2n(CCCOC)nnn2)NCC(Cl)Cl)c(Cl)ncn1C C12(OCC)CCC(C(=O)NC3CCN(c4sccc4C(=O)OC)C3=O)(CC1)C2 CC1CN(C(=O)CC2C3CCCC3N2C(C2CCS2(=O)=O)=O)c2cccnc21 C1(NC(C2CC3CCC2C3)=O)CCCN(CC(=O)NC(c2c(C)onc2)=O)C1 N1(c2nnc(CC)s2)CCCC(NC(C2CCC(OC(C)C)CC2)=O)C1C N1(C(C(C)NS(CC)(=O)=O)=O)CCCN(C(=O)Cc2ccc(Cl)nc2)CCC1 Cn1ccc(C=CC(N2CC(O)CC2CNC(c2cccc(OC(F)F)n2)=O)=O)c1 c1(C(=O)NC2C3N(C(C(C)(C)CO)=O)C(CC3)C2)cc2ccccc2nn1 c1(C(=O)NCCOC2CCN(C(C3CC3[N+](=O)[O-])=O)CC2)cc2n(n1)CCCO2 C12CC3(CN1OC(=O)C14CC(C(C)N1C2=O)C4)CC3(F)F.c1(CN)ccccc1 CC(C)C(C(=O)NCc1ccc(SC(C)C)nc1)c1cnn(C)c1.C12CC1(O)C2 C1(C)(CC(=O)NCC(N2CCCC2)C)CCN1C(=O)Cc1ccco1 C1(NC(C(c2cnn(C)c2)OC)=O)CC2CC(C1)N(CC1CCCC1)C2 C1(C)(C(=O)NC(C(C)C)CNC(C2CCS(=O)(=O)C2)=O)CCN(C)CC1 c1(C(=O)NC2C(CNC(C(n3ccc(C)n3)C)=O)CC2)ccc2scnc2c1 c1(C(=O)NC(CN(C(=O)CC2(c3ccon3)CC2)CC)C)nc[nH]c2nccc1-2 Cc1nc(S(=O)(=O)NCC(=O)NC2CN(C(=O)C(C)(F)F)CCC2(C)C)cn1C c1(CC)ccc(F)c(CN(C=O)CC2(c3cc(Cl)cc(Cl)c3)CC2)c1 CC(C)C(C)C(=O)N1CC(N(C)C(c2ccc(N(C)C)cc2)=O)C1 N1(C(CCOC2CN(C(C=CCOC)=O)C2)=O)CC2COCC2(CO)C1 C=C1CCC(C(=O)NC2C=CC(CC(=O)NC3(C)CC(F)(F)C3)C2)CC1 C1(NC(c2c(Cl)cc(C)s2)=O)CC2CN(C(c3ccc(N)cc3O)=O)CC2C1 c1(CC)ncccc1C(=O)NCC(CCCC)NC(=O)COC(C)(C)CC C1(C(=O)NCCCN(C(=O)CC2CCC23CCC3)CC)(N(C)C)CCCOC1 N1(C(=O)NC(c2cnn(CCc3ccccc3)c2)C)CC(O)C(O)C12CCCC2 C(=O)(CCC(C)(C)C)NCCN(C(=O)CCC1C(=O)ON=C1C)CCOC N1(C(C(COC)Cl)=O)CC(NC(c2ccc(Br)cc2Br)=O)C2(CC2)C1 C12(CCCCC1)CNC2.N12CC(OC)(C1)C2=O.c1(C(=O)NC)nc(C(N)=O)co1 N1(C(C(C)CO)=O)CC2(CCN(C(=O)Cc3c(Cl)cnn3C)CC2)CC1C C=C1CCN(C(c2cc(C(N)=O)co2)=O)C(C(=O)NCCCC2CCCCO2)C1 c1(CN2CCC(n3cc(C(N)=O)nn3)CC2)cc(F)cc(Cl)c1 c1(OC)ccc(C(N2CCCC(NC(c3ncn(C)n3)=O)C2C)=O)cc1Cl C(CCC(F)(F)F)(C(=O)NCc1ccc(-c2ccccc2)cc1F)OC C1(NC(c2n(CCC)ccc2)=O)CN(C(=O)C(C)Oc2ccccn2)CCC1C c1(OC)cc(OC)nc(N2CC(CNC(=O)CCC3CC3(Cl)Cl)CC2C)n1 C=CCC(C)(C)C(=O)N1CCC(C)(CNC(=O)C(c2ccc(F)cc2)C2CC2)C1 c1(C(=O)NC(C2CCN(C(CNC(C)=O)=O)C2)C)cnc2ncnn2c1C(C)C C(=O)(CCC(CC)NC(=O)CC1CCC(=O)C1C)N1CCC(C(C#C)C)CC1 C(=O)(C1=C(Cl)CCC(C)C1)NCCCC(C)NC(CCC(=O)NCCC)=O C(O)(C(F)(F)F)C1(CC(=O)NC2CN(C(C=C(C)C(F)F)=O)C2)CCC1 CN1CCOC(C(=O)NCC2(O)CCN(C(C3(C(F)(F)F)CCCC3)=O)C2)C1=O Cc1c(N(C(c2ccnc(Cl)c2)C(=O)NCC(C)C)C)cccc1Cl CC(O)CCN=c1[nH]c(=NC2CCC(N3CCCCC3)C2)c2c(F)cccc2[nH]1 N1(C(c2cc(C(N)=O)oc2)=O)CC2(CCN(C(C3CCC(C(F)(F)F)O3)=O)C2)C1 C1(C(=O)Nc2ncc(C)c(Br)c2)CC12CCN(C(=O)C(C)n1ccnn1)CC2 C1(C(=O)OC)CN(S(C)(=O)=NC(=O)C(c2ccccc2)OC(C)(C)C)CCO1 C1(OC)CC(CNC(c2cc(C)c(Cl)s2)=O)N(C(C2CCN(C)C2)=O)C1 C1(CNC(c2nnc(C)s2)=O)CC2(CCN(C(c3ccc(=N)[nH]c3)=O)C2)CO1 n1(CC)ccc(=NC(=O)C(C)(C)C2CCCN2C(=O)Cc2ccnn2C)[nH]1 Nc1cc(F)c(O)cc1C(N1CCCC(C2CCCCN2C(=O)CNC=O)C1)=O c1(C(=O)NC(CNC(CC(CCC)O)=O)C)ccc2nc(O)[nH]c2c1F c1(C(=O)NC2C(CNC(C(C)OC)=O)C2)cnc(C)nc1C1CC1 Cn1cc(CN2CC(=O)N(CCCc3cc(F)cc(F)c3)C2=O)c2ccccc12 c1(N2C(=O)CCC2)ccc(S(=O)(=O)NC2CCCCC2C2CCCCO2)cc1 n1(CC)nc(C(=O)NCC2CCC(CNC(=O)COC3CC3)CC2)ccc1=O C1(C(=O)NC(C)CN(C)C(c2c[nH]nc2C2CC2)=O)CCC(C)(C)CO1 CC1(C)CC(C(=O)NC2CCCN(C(=O)Cn3cnnc3)C2)CC(C)(C)S1 c1(C(N2CC(C)C(NC(C3CCSCC3)=O)CC2)=O)ccc2cccnn12 Cc1c(CC(=O)NCC2(NC(=O)CC3CC=CCC3)CCC2)ncn1C C(=O)(C(C(C)(C)C)NC(=O)CC1CCOC1)NCC1(C)N=C(C)SC1 c1(C(=O)NCc2occ(C(=O)Nc3ccc(C#C)nc3)n2)cnc(C)c(C#N)c1 Cc1cc2c(NCC3(C)CCNC3)ncnc2[nH]1.C1(C(=O)N)(CN)CC1 C1(CNC(C2N(CC)CCCC2)=O)CC2(CO1)CN(C(=O)C(CC)(CC)CO)C2 C1(NC(=O)CCOC2CCCCC2)CCCC12CN(C(c1cn[nH]c1)=O)C2 c1(C(C)OC(COCCCCOC)=O)nc(-c2ccccc2)no1 C(C(C)(Cn1cccn1)NC(c1n[nH]cc1Cl)=O)NC(CC1CC(C)C1)=O Cc1[nH]nc2ncnc(N3CCCC3(C)CNC(c3ncoc3C3CCC3)=O)c12 c1(C(=O)NC(C)C(CO)NC(c2nccnc2N)=O)ccc2nonc2c1 C1(CC(C)C)CCN(C(=O)C(C)N(C(=O)C(C2CCCCC2)F)C)C1 N1(C(Cc2c(C)ncs2)=O)CCC(n2cc(CNC(=O)C(C)N(C)C)nn2)CC1 C1(CC(=O)NC(C(C)O)C(=O)OC(C)(C)C)(C(F)(F)F)CC(=O)N(O)C1 C1(C(=O)NC(C)CNC(=O)CC=CCN2CCCC2)COC(=O)N1C C1(C(=O)OCC)Cc2cc(S(=O)(=O)N3CC(N4CCOCC4)C(C)C3)ccc2O1 C(C)(CCN=c1nc(OCC(C)C)cc[nH]1)NC(C1(C)ON=C(C)C1)=O CCC(CN(C)C)CC(=O)NCC1CC(OC)CN1C(C1CN(C(C)C)C1)=O C1(C(=O)NC2C(CN(C)C)CCC2)CCOCCN1C(=O)CCCF N1(C(CC2N(C(c3cnn(C(C)C)n3)=O)CC(F)C2)=O)CCCC(CO)CC1 N1(C(c2ccc(C)cc2C)=O)CCC2(CC1)CC2NC(c1cc(Br)no1)=O CN1CCN(CC(N2CCC(OCCCC(F)(F)F)C2)=O)CC1 C(=O)(C#CC1CCC1)NC(C1(O)CCN(C(c2ccc(C#N)cc2)=O)C1)C c1(OCC)ccc(CCC(=O)NCC(C2CC2)NC(C2CC23CC3)=O)cc1 CCC(C)(COC)C(=O)NOCC(=O)Nc1conc1C(C)C C1(CNC(CC2(OC)CN(C(C3C(OC)CCCC3)=O)C2)=O)CC(C)(C)CCO1 O=C(CCC(F)(F)C(F)(F)F)NC1CN(C(=O)CC23CCOC2CCOC3)C1 c1(NC(C2(NC(C3CC4(CC4)CO3)=O)CC(F)(F)C2)=O)ccc(O)c(F)c1 N1(Cc2cn(CCC(=O)NCCSC)nn2)CCCCC1C1CC1.CCO CS(=O)(=O)C1(C(N2CCC(Oc3ncccc3F)CC2)=O)CCNC1 N1(C(c2oc(C(=O)OC)c(C)c2)=O)CC2CCC2(CNC(C2(C)CC(C)C2)=O)C1 CCC(F)(C(=O)OC)C(=O)N1C2CCC1C(CNC(=O)COc1cccnc1)C2 CC1(CNC(C2CCCCC2O)=O)CC(F)(F)CN1C(=O)C=Cc1ccccc1 C1(C(N(CC(C)O)CCNC(C23CC(C)(CCO2)C3)=O)=O)CCCCN(C)C1=O C1(NC(Cc2c(C)non2)=O)CCCC(CNC(=O)CCCN(C)C)C1 N1(C(c2ccc3cccnn23)=O)CCC2(CCCN2C(C2CCCS2)=O)C1 c1(OC)cc(C)[nH]c(=NCC2CCCN2C(c2cc(C3CC3)[nH]n2)=O)n1 N1(C(CC(=O)NCC#C)=O)CCN(C(=O)CO)CC1C C1(C(=O)NC2C(CNC(Cc3c(C)scc3)=O)COC2)Cc2ccccc2S1 Cc1cc(C(=O)NCCC(C)N(C)C(c2cc(CO)n(C)n2)=O)cnc1O c1(N2CCC(C)(NC(C(C3CCCOC3)OC)=O)C2)ccncc1C#N CCC(CC)CC(=O)N1CCN(C(C2CCCC(N(C)C)C2)=O)C(C)C1 c1(CC)[nH]nc(C(=O)NCc2cn(C)nn2)c1[N+](=O)[O-] c1(OC)cc(C(N2CCC(NC(=O)CCn3cc(C)cn3)C(F)C2)=O)ccc1F N1(CCNC(C2N(C(Cc3n(C)nnc3)=O)CC2)=O)CCCCC1=O C1(C(=O)NCC2(CCNC(C3(OC)CCOC3)=O)CC2)CCc2nnnn2CC1 N1(C(CCNC(=O)OCC)=O)CC=C(C(=O)NC2(C(=O)OC)CC2)C1 c1(OC(C)C)cc(C(F)(F)F)cc(CNC(N)=O)c1.C12CCCN1C(=O)C(C)S2 Cn1cc(C(=O)NCC2(NC(c3ccnc(C(F)(F)F)n3)=O)CCC2)cc1Br Cc1cc(C(=O)NCCCN2CCCC(C(N)=O)C2)nn1C1CCC1 C1(C(=O)NC)CCCC(C#N)C1.c1(C(C2(CC)CC2)=O)ncc[nH]1 c1(C(=O)NCC2(F)CN(C(C3C(C=C)C3)=O)C2)ccc(C)c(Br)c1C c1(NC(C2CC3CNCC23)=O)cccc([N+](=O)[O-])c1 C12(C(=O)NCC(C(C)C)N(C)C)C(NC(c3ccncc3Cl)=O)C3CC1C2C3 n1(CC(=O)NC(CC=C)CNC(C2CC(=O)NC2(C)C)=O)c([N+](=O)[O-])cnc1C C1(CCOC)(NC(c2cnccc2C)=O)CCN(C(c2nocc2Cl)=O)C1 Cc1c(OCC(N2CCOCC2CCNC(=O)CCC(C)(C)F)=O)cccc1Cl N1(C(C(=O)NCC(F)(F)F)=O)CCC2(CC1)CC2C(=O)NC1CCCC1C1CC1 c1(C(=O)NCCC2CCN(C(C(CO)NC(N)=O)=O)C2)cncc(CO)c1 c1(C(N(CC(C)N(C(CCCC=C)=O)C)C)=O)ccc2c(c1F)CCC2 C1(CCNC(=O)COCCCF)CN(C(=O)Cc2cccc(Cl)c2)CCO1 c1(CN(CCCOC)CC(=O)OC(=O)Cn2ccccc2=O)ccc(C)cc1Br N1(C(c2c(Br)ccc(C)n2)=O)CC2CCC1CN2C(=O)CC(O)C(C)C C1(NC(C(C(C)C)n2ccc(C)c2)=O)CCC2(CC1)CN(Cc1ccccc1)C2 C1(NC(C(CCC)O)=O)CN(C(c2ccc(-n3cncn3)c(N)c2)=O)C(C)(C)C1 N1(C(CCCCCC)=O)CCCC2CN(C(=O)CNc3ccc(O)cc3)CCC12 c1(N(CCCOCC)C)nc(=NC(C)c2ncccc2C)[nH]c2cccnc12 Cc1nc(Cl)ccc1CC(=O)NC(C1CCCC1)CNC(=O)CCCNC(N)=O N1(C(C=C2CCC(C)CC2)=O)CCCC(F)(CNC(=O)CC23CC(C2)C3)C1 c1(CC(=O)NC(CC=C)CN(C(=O)CCC(=C)C)CC)coc2cc(O)ccc12 C1(C)(C(=O)NC)CCCN1C(=O)CC1CCN(C(c2cn[nH]c2)=O)C1 CC(CN=c1[nH]c2c(c(=NCC3COC(=O)N3)[nH]1)COCC2)C1CCC1 N1(CCNC(=O)CC2CC2C2CCCC2)CCN(C(C2CCNC(=O)C2)=O)CC1 Cc1ccc(Cl)c(C(=O)NC(C2(O)CCN(C(=O)C(C)C#N)C2)C)c1 C=CC1COCCN1C(=O)CCC1CC(NC(C2CCCC(O)C2)=O)C1 c1(C(=O)NC2(CCCC)CC2)cc(CNC(=O)C=CCN2CCC2)nn1C c1(NC)ncccc1C(=O)NCc1c[nH]nc1C(N1CC(C)C(O)C1)=O C(C(O)CCCC)NC(C(C1(O)CN(C(CCOCC#C)=O)C1)F)=O C1(NC(c2n(CC)ncn2)=O)CCC(C)(CNC(c2ncccc2CO)=O)CC1 c1(OCCONC(c2[nH]cc(CC)n2)=O)ccc(Cl)cc1C.C12CCC1C(=O)N2 CC(C)(CCNC(C1CC(N(C)C)C1)=O)NC(=O)CC1CCC(O)C1 C1(C)(CC)CCCN(C(C2CN(C(c3ccc(C)cc3OC)=O)CCO2)=O)CC1 C1(C)(C(N(c2cccc(C#N)c2)C)=O)CC(O)CN1C(=O)C1=C(Cl)CCC1 N1(CCC)CC(N=c2ccn3ncc(S(=O)(=O)N4CCSC(C)CC4)c3[nH]2)C1 CC1CCC(C(N2CCC(C)(CNC(c3ccc(C(F)(F)F)[nH]3)=O)C2)=O)CC1 C12(NC(c3c(C)nc(C4CCCCC4)s3)=O)CCN(C(=O)C3=NOCC3)CC1C2 C(=O)(C#CC1CCC1)N1C(CNC(C2C(C)(C)CCO2)=O)CCCC1 c1(C(=O)NCC2CN(C(c3ccc(C)cc3)=O)C(C)CC2)cccc2nn[nH]c12 C1(c2ccccc2)(NC(C(C)N2CCC2)=O)CN(C(=O)CC2CC2C)C1 C(CN=c1ccc(C#N)c(CC(C)CS(C)(=O)=O)[nH]1)=CCCC CC1C(NC(=O)C(C)(C)C)CCN1C(=O)Cn1ncccc1=O C1(C(C(=O)NCc2ccc(CC)s2)(C)C)CCCN(C(=O)C=CCO)C1 C(=O)(C1=CCCC1(C)C)NCC1C(NC(CC2(NC(C)=O)CC2)=O)CCO1 C1(C(N2CC(NC(c3cn(C)nc3OCC(F)F)=O)C2)=O)CC(=O)NC(=O)C1 c1(C(=O)NC2CC(CNC(Cn3c(C)nnn3)=O)C2)cn(CC(F)(F)F)nc1C c1(CC(=O)NC2(CO)CN(C(CCOCCCC)=O)C2)ccc(C)c(F)c1F Cc1onc(O)c1C(=O)NC(C)CNC(c1nccn1C(C)C)=O N1(C(C2C(CC)CCC2)=O)CCC(C)(NC(c2cnc(Cl)s2)=O)C1 C(=O)(C(CCF)NC(c1cc(OC)n[nH]1)=O)NC(C#C)CC c1(C(C(=O)N(CC(O)CNC(c2cn(C)nc2Cl)=O)C)(F)F)cccc(Cl)c1F N1(C(CCC#C)=O)CCCOC(CNC(c2ccnc(-c3cccnc3)n2)=O)C1 Cn1nc(C(=O)NC2CC(CCC(=O)Nc3ccc(O)nc3)C2)ccc1=O S(=O)(=O)(c1ccc(NCc2csnn2)c(Cl)c1)N1CC(CCOC)OCC1 N1(C(c2cncc(OC)c2)=O)CCC(NC(C2CNC(=O)N2C)=O)CC(O)C1 C(=O)(CC1(O)CCOc2ccccc21)NC1CN(C(c2c(C)ncc(Cl)c2)=O)C1 CCC(F)(F)C(C)(C)NC(C1C=CCN(C(c2cccc(F)c2N)=O)C1)=O Cn1nc(C(=O)Nc2cc([N+](=O)[O-])c[nH]2)c2c1CCN(c1nnc(C(F)(F)F)s1)C2 N1(C(c2c(OC)cncc2)=O)CCC(C)C(NC(=O)CN2CCC2)C1 N1(C(CCc2c(C)cccn2)=O)CC(CNC(C2(F)CCC2)=O)C(C)(C)C1 N1(C(C(C(C)C)(C)C)=O)CC(CNC(C2(C)CCCNC2=O)=O)C2(CCC2)C1 C=C(C)c1cn(CCC(=O)N(CC)Cc2coc(-c3ccc(Cl)cc3)n2)nn1 c1(C(=O)NC2CN(C(c3cc(C)nc(C)c3)=O)CC2C)cccn2ccnc12 c1(C(=O)NC2CCN(C(=O)C(c3ccccc3)O)CC2)cnc2[nH]c(O)nc2c1 CC1(NC(c2cncnc2)=O)CCCCC1C(N1CC2(CC2)C1)=O C(C)(CNC(=O)C(=O)NC(C)C)(C(C)C)NC(C(c1ccc(OC)cc1)CC)=O c1(C(N2C(C(C)C)C(NC(C3CC3[N+](=O)[O-])=O)CC2)=O)ccnc2c1CCC2 N1(C(c2c(CC)cco2)=O)CC(F)(F)CC1CNC(=O)CCc1nc(C)c(C)[nH]1 c1(NC(c2c(-c3cc(C)ncc3)c[nH]n2)=O)cc([N+](=O)[O-])c(F)cc1F C(=O)(C(C)S(N)(=O)=O)NC(C1CN(c2cc(CC3CC3)ncn2)CCO1)C O(NC(=O)C(Cc1ccoc1)NC(C1CN2CCC1C2)=O)CCC(C)C C(=O)(C(O)CC(F)(F)F)N1CC(N(C(CC(C)=C(C)C)=O)C)C(O)CC1 C1(NC(C=CCN(C(c2cc(CCC)on2)=O)C)=O)CN(C)NC1=O c1(C(N(CCc2cn(-c3ccc(OC)cc3)nn2)C)=O)cc2ccccc2cn1 C(=O)(CCCCCF)NCCNC(c1cc(C(N(CC#C)C)=O)no1)=O c1(OC)cccc(C(=O)NCCC23CCC(C2)N(C(=O)CCNC(C)=O)C3)c1N C(=O)(C(F)(CNC(=O)C(C)C(F)(F)F)C(C)C)NCc1ncc(CC)s1 CCC(C(=O)NC(C1(O)CCN(C(=O)CCCSC)CC1)C)C(C)C S(=O)(=O)(c1cc(C(=O)NCC2CN(C(c3cc(C)[nH]n3)=O)C2)c(C)o1)NC N1(C(CCCCC=C)=O)CCN(C(C2CCCCN2CCC)=O)C2COCC12 C1(NC(c2c(C)cc(C)s2)=O)CN(C(=O)C(C)N=[N+]=[N-])CC12CCC2 Cc1[nH]nc2ncc(C(N3CCCCC3CNC(C3(C)CCCCC3)=O)=O)cc12 c1(N(C(C)=O)C)cc(F)c(F)cc1Br.c12c(C)[nH]c(c1C)C(=O)C(C#N)C2=O c1(C(N(CC(C)(C)NC(c2cc(C)c(O)nc2)=O)C)=O)c(F)ccc(F)c1Cl c1(N(C)CC23CCCC2OCC3)nc(C)cc(=NCC2CNC(=O)CO2)[nH]1 C1(CNC(C(C)SCC)=O)CN(C(=O)CC2CCC3CC23)CCCO1 C1(CNC(=O)COc2ccon2)CC12CCN(C(c1cnc(O)s1)=O)CC2 C1(COC)(CNC(c2cc(OC)ns2)=O)CCCN1C(C1C2CCC(=O)C12)=O N1(C(CNC(CCC)=O)=O)CC2CC(NC(C3CCC(=O)N3)=O)CC2C1 C(=O)(C(C)(CC)C(=O)NC1CC(CNC(=O)Cc2cc(F)cc(Cl)c2)C1)OCC C(=O)(CCCN=[N+]=[N-])N1C(CN(C(C=C(C)Cl)=O)C)CCCC1 C12(C(=O)NC(C3CCN(C(=O)CCC(N)=O)C3)C)CCC(C)(C1)OC2 C1(NC(=O)C(O)Cc2cnc[nH]2)CCOC12CCN(C(=O)C(F)F)CC2 c1(CC)c[nH]c2ncnc(N3CCCC(NC(c4oc(CC)nc4C)=O)C3C)c12 C=CCC1CNC(=O)C2CC2NC(=O)C2(CC2)OCC(=O)N1.C(C(C)(C)C)OC C1(C(N(CCOC)CCF)=O)C2CC(O)C(C2)N1C(c1ccns1)=O CCCCC(O)C(=O)N(C)CCNC(C1(F)CC1(F)F)=O CCC(C)C(O)CC(=O)NC1CC(Cn2cc(CCCCCCO)nn2)C1 Cc1oc(C#N)cc1C(=O)NC(Cc1cnc[nH]1)C(=O)NC1(c2nc[nH]n2)CC1 c1(OCC(N2CC(NC(c3c(CC)c[nH]c3)=O)C(C)C2)=O)ccc(Cl)cc1CO c1(C(=O)NC2CCCCC2NC(c2cccn2C2CC2)=O)ccc2c(c1)CCN2 CCCC(C)CCCC(=O)N1CC(NC(c2ccnc3c2CCC3)=O)C(C)(C)C1 Cc1nnc2n1CCN(C(C1(C)CCCN1C(c1ccc(Cl)c(O)c1)=O)=O)C2 c1(C(N2CC(CNC(CCCCCC)=O)OCC2)=O)cc2n(n1)CCOC2 Cc1c(Br)cc(C(N2C3CCC(C3)C2C(=O)NC2CC(F)(F)C2)=O)cc1Br C1(NC(c2n(CC)ncn2)=O)CC2(CCN(C(=O)C(O)CC(C)C)C2)C1 Cc1nn(C)c(C)c1CC(=O)NC1CC(N(C)C(C2C=CCCC2)=O)C1 C(=O)(C1c2c[nH]nc2CN1C(=O)CCc1ccco1)N(C)CCOCCCO C1(NC(CNC(NCC)=S)=O)CC2CCCC(C1)N2C(c1c(I)ccnc1F)=O Cc1c(C(=O)NCCNC(=O)C(C)(C)N(S(C)(=O)=O)C)cccc1F N1(CC(=O)NCC(C)CN(C(=O)CN2CCSCC2)C)CCC(CO)CC1 C(=O)(C(C)CCN1CCOCC1)NCC1(C(=O)NCCN(CC)CC)CC(=C)C1 N1(C(C(CC)NC(=O)OC(C)(C)C)=O)CCN(C(C23CCC2C3)=O)CC1COC C1(CC(=O)NCC(N2CCOCC2)C2CC2)C=CCCC1 c1(C(N2C(CCNC(C3CC(C)OCC3)=O)CCCC2)=O)ccc2c(c1)CC2 C1(N(C)C)CN(C(=O)CCOCC2CC2)CC1CNC(=O)Cn1ccnn1 c1(C(N(CCCN(C(CC(COC)C)=O)C)C)=O)cnc(C2CCCC2)[nH]c1=N C1(NC(C2N(CC)CCC2)=O)CCN(C(c2ccccc2OC)=O)C(C2CC2)C1 CCCC(CC)CCC(=O)N1CCC(C2(C)CC2)C1 C(=O)(C(CCCOC)N(C(=O)Cc1cccs1)C1CC1)NC(C#C)(C)C C(=O)(C1(C)CCn2ccnc21)N1CC2(CCN(C(C3C(C(=O)OC)C3)=O)C2)C1 C(=O)(C1=NOC2COCC12)NCCCCCNC(=O)CSc1cn[nH]c1 c1(C(N)=O)cc(F)ccc1C(=O)NCC1CCN1C(C1(C2CCCCO2)CC1)=O c1(CC)nccn1C(C)CC(=O)NCCCCNC(C1CC1F)=O c1(C(=O)NC(c2cccnc2)C(=O)NCCc2c(C)ncs2)csc(C#N)c1 C1(NC(c2c(CC)ocn2)=O)C2CC3C(C2)C13C(=O)NCC1C(C)C1C C12(C(N3CCC(NC(CCC(CC)C)=O)(CC)CC3)=O)CC1Cc1c[nH]nc12 N1(C(=O)C(F)n2ccnc2)CC23CCCC2(C1)CN(C(C12CC1C2)=O)C3 CC1COC2(CCN(C(c3cncs3)C(=O)Nc3ccc(Cl)cc3F)CC2)O1 CC(C(=O)NCC(C1CC1)NC(c1cc(O)nn1-c1ccccc1F)=O)C(F)F C(=O)(C(F)(F)C(F)(F)F)NC(C(C(C)C)C)CNC(C1(C2CCC2)CCC1)=O c1(OCC=C)c(C(=O)NCC(C)(O)CNC(=O)C(C)SC(C)C)cccc1C c1(OCC(=O)NCCCCCNC(c2cnc(C)n2C)=O)cccc(F)c1F Cc1ccc2[nH]nc(C(=O)NC3CCN(C(=O)C(C)n4ccnc4)CC3O)c2c1 n1(CC(=O)NCCC2N(C(C3C(C)C3(F)F)=O)CCC2)ncn2cccc2c1=O N1(C(C(CC)Br)=O)CCC(N2CCC(=O)CC2)C2(CC2)C1 C12(NC(CCCc3onc(C)n3)=O)CCC1CN(C(c1cccc(C)c1O)=O)C2 CC1CN(C(=O)CCc2ccc(CO)cc2)CCC1NC(C1C2CCC1CC2)=O C1(C(=O)NC(C2CC=CCC2)C(=O)NCCn2c(CC)nnc2)CC(C)CCO1 CC1(C)CC(O)(C(N2CC(CNC(c3ccc(C(F)(F)F)cc3)=O)C2)=O)C1 Cc1nc(C(=O)NC2CCCN(C(c3cccc(C(=O)C4CC4)c3)=O)C2)c(C)s1 C1(C(=O)NCC(C)(C)OCCNC(c2conc2C(C)(C)C)=O)CCCC1O N1(c2ccc(NC(N3CCC(NC(CC#N)=O)C3)=O)cn2)CCS(=O)(=O)CC1 C=CCC(CC=C)C(=O)N1CCC(CCC(=O)N(CC(O)C(F)(F)F)C)C1 CC1CC(NC(c2cn(C3CCOC3)cn2)=O)CCN1C(=O)C1=CCSC1 N1(C(C(CC=C)OC)=O)CC(C(N2CCC3CCCC23)=O)CC(C)(C)C1 C1(O)(C(C)(C)NC(C)=O)CCN(C(=O)CN(CCO)CCO)CC1 C(=O)(C(O)C(C)SC)N(CCC)CCNC(=O)Cn1ccc(C)n1 n1(CC=C)cc(C(=O)NC(CO)C(=O)NCC2(O)CSC2)cn1 C1(NC(C(C)(C)C#N)=O)CC2CCCC(C1)C2NC(C1CC12CCSCC2)=O C(CN=c1nc(C(C)(C)C)[nH]s1)(CC(C)C)NC(Cc1c(C)ccs1)=O c1(C(c2n(CCCC)nnn2)NC2CC(F)(F)C2)cnc(OCC)c(C)c1 C#CCCCC(C)C(=O)NCCC1CC(NC(=O)COCC2CCCOC2)C1 c1(C(=O)OCc2nc(C(C)C)on2)ccc(S(=O)(=O)O)cc1 c1(C(=O)NC(C2CCN(C(CN(CCC)C)=O)C2)C)cc(SC)ccc1[N+](=O)[O-] C12(CC(O)C1)C(=O)N2.C1(CNC(C)=O)(NC(=O)CC2(N(C)C)CC2)CCOC1 N1(C(c2c(CC)oc(C)c2)=O)CCC(NC(c2cc(CO)oc2C)=O)C(F)C1 c1nnc(S)s1.C1CC(=O)N1.C1C(OC)CNC(=O)C1.C(=O)(NCC)OC C(=O)(CC(C)(C)C(F)(F)F)NCC1CC(CNC(CCC(=O)OCC)=O)OC1 N1(C(C(n2ccc(C)n2)C)=O)CCN(C(c2ccc(C)o2)=O)C(C2CCC2)C1 C1(C(N(C2CCCC2)CC(C)O)=O)CCC(NC(c2ccccc2)=O)CC1 c1(OC)cnc(F)c(C(=O)NCCC2(O)CN(C(=O)CCn3cc(C)cn3)C2)c1 N1(C(C2N(C)C(=O)CC2)=O)CCC2(CC1)CC2(C)C(=O)NCC1CCC(=O)N1 c1(Cn2c(-c3c(-c4c(C)cc(F)cc4C)csc3)ncc2)ccc2ccccc2n1 C1(NC(c2[nH]c(=NCc3c(OC)ncc(Br)c3)sc2)=O)CCC2(CC1)OCCO2 C1(CNC(C(F)=CCC)=O)CN(C(=O)C(c2ccccc2)F)C(C)(C)C1 c1(CNC(C)C(O)C(F)F)ccc(F)c2cccnc12 N1(C(C(=O)NC(C(=O)OC)C)C2=NOC3CC23)c2ccc(Br)cc2CC1C c1(NC(c2ccc(F)cc2)CC)ncccc1S(=O)(=O)NC(C1CC1(C)C)CC C1(C(C)C)CN(C(c2ncn(C)n2)=O)CCC1NC(c1c[nH]cc1C1CC1)=O C(=O)(CCCCCF)N1CCC(CN(C(c2c(OCC)oc(C)n2)=O)C)CC1 N1(C(CC(=O)N(C)C)=O)CC(NC(c2c(Cl)ccc(Cl)c2O)=O)CC2(CC2)C1 c1(C(=O)NCC(CC)Nc2ccnc(C(F)(F)F)n2)ccnc2ccnn12 C(=O)(C#CC1CCCC1)NCC(CN(C)C(c1ncnc2ccsc12)=O)O c1(C(N2C(C)CC(NC(CC(CC)(F)F)=O)C2)=O)cncc2cnccc12 N1(C(c2cnn(CC(F)(F)F)c2)C(=O)NC2(C)CC2)CCc2c(Cl)cccc21 c1(C(N2CC(CNC(C(Cc3cccc(OC)c3)=O)=O)C2)=O)cccc(O)c1C c1(OCC)ccc(S(=O)(=O)N(CC(c2cccc(C(F)(F)F)c2)O)C)cc1OC C#CC1(C(=O)NCCCC(CO)NC(C2CC(C)(C)C2)=O)CCCC1 C1(C(=O)NC2C=CCN(C(c3ccc(C#N)s3)=O)C2)CC12CCS(=O)(=O)CC2 CC(C)S(=O)(=O)c1ccc(CC(=O)NC2CN(C(=O)C(F)C(C)(C)O)C2)cc1 C=CC1COCCN1C(=O)C(CC)NC(=O)OC(C)(C)C.C12CC1CNC(=O)N2 C1(NC(C2(CC)CCCC2)=O)CCCCN(C(c2cnncc2C)=O)C1 Cc1onc(C2CC2)c1C(N1CCCCC1CNC(c1ccnn1C1CC1)=O)=O CCC(C(=O)OC)C(=O)NC(C)(CNC(C12CCCC1CCC2)=O)C1CCC1 Cc1cc(N)c(C(=O)NCC2(CCNC(=O)CO)CC2)cc1F c1(OCC)cc(C(=O)Nc2ccc(C(N3CCC(CF)CC3)=O)nc2)ccc1Br CCCCC(O)CC(=O)NCc1csc(CNC(=O)C(c2ccccc2F)C)n1 c1(CN(C(=O)CCCn2cc(-c3cnn(C)c3Cl)nn2)CC)ccccc1OCC C1(NC(CN2CC(=O)NC2=O)=O)CCN(C(C2(C(F)(F)F)CC(O)C2)=O)CC1O c1(C(=O)NCC(C)NC(CCc2onc(C(C)OCC)n2)=O)cc(N)ccc1F Cc1c2c(nn1C)CCC(NC(=O)CCCCCn1cc(C3CCCO3)nn1)C2 N1(C(C(c2ccc(Cl)cc2)C)=O)CCCC(O)(CNC(=O)C(C)(C)N(C)C)C1 C(=O)(CC1c2ccccc2C(=O)N1C)NCCC1(NC(C(C)CC2CC2)=O)CC1 c1(C(C)N(C)CCC2CCN(C(C3CCCOC3C)=O)CC2)ccc(Cl)nc1 S(=O)(=O)(c1ccc2c(c1)CCO2)N(C1CCNCC12CC2)Cc1n(C)ncc1 N1(C(CN(C(CC2CC(SC)C2)=O)C2CC2)=O)CCC(O)C(C)(C)C1 N1(Cc2c(C(=O)O)cccc2)Cc2[nH][nH]c(=NC(=O)C(F)(F)Cl)c2C1 C(=O)(CCC(C)CN(C)C)N(CC(C)(C)CCC)C(C1C2COCC12)=O C12(CNC(C3CC(C(=O)OC)C3)=O)CCCC1N(C(=O)CCCCC)CC2 c1(C(N2C(CNC(c3ccnn3-c3ccncc3)=O)CC2)=O)c(Cl)nsc1Cl CC(=O)C(C)CC(C)C(=O)N1CC(C2CC2C(=O)NC2CC2CC(C)C)C1 C1(CC(=O)N(CC(C)C(=O)N(C2(CO)CC2)C)C)CCCC2CC12 c1(CC)cccc(C(=O)NC2CCCCC2NC(C2(C)CC=CCC2)=O)n1 C12(C(=O)NCCSCCC=C)CC1CCN2C(=O)C(C)SC(C)C N(C1CCC(C)(C)c2ccccc21)c1c(C(C)O)cncn1 C(CCC(C)C(=O)N1CCOC(CN(C(=O)Cc2cc(C)cc(C)c2)C)C1)OC C(C)(COCC)(C(N)=O)NC(C(Cn1cncn1)NC(CC)=O)=O c1(CC)cc(C(N2CC(F)(CNC(=O)CCc3ccc(C)s3)C2)=O)nn1CCO c1(N(C(C)(C)C)C(=O)CONC(C2CC3CC3C2)=O)ccc(Cl)c(C#N)n1 C12(OC)COC(C1)C(NC(=O)COC1CCN(C(c3sc(C)cc3C)=O)C1)C2 C1(C(N2CC(C(=O)NCCc3cn(C)cn3)(COC)C2)=O)CCCCC1(C)C N1(C(c2ccc(OC)nc2Br)=O)CCC(C2CCCNC2)C1 CCC(CC)C(=O)NC1CCC(CNC(=O)Cc2ccc(C)nc2)C1 c1(C(C(=O)NCC2CCOC2)N(C2(COC)CCC2)C)cccc([N+](=O)[O-])c1C CN1CCC(CCn2nnnc2N2CCC(C3CCCO3)CC2)CC1 C(C(C)(O)C(=O)NCC1CCCN(C(C2CN(C3CCOC3)C2)=O)C1)OC c1(CC(=O)NCC(CNC(Cc2cc(C)no2)=O)F)c(C)cccc1F c1(C(O)CNCc2ncccc2Br)cccc(C(F)(F)F)c1 Cc1cc(=NCCCn2cc(Br)cn2)[nH]c(NC2CCc3n[nH]cc3C2)n1 C1(C(=O)NC2CCC(F)CC2)(CNC(C(SC)SC)=O)CC2(CC2)C1 CCC(CC)(CCNC(=O)Cc1cscn1)NC(c1cc(CCCO)on1)=O CC(CC(=O)NC1(CF)CCN(C(C23CCC(CC2)C(C)O3)=O)C1)C(F)(F)F c1(CC)ccc(C(=O)NCC2CC(NC(c3ccncc3F)=O)C2(C)C)cc1Cl c1(COC)cccc(C(N2CC(NC(C3(C)CCCO3)=O)CC2C)=O)n1 N1(C(c2c(OC)ccnc2)=O)CC2(CCCC2)C1C(N1CC(C(N)=O)C(C)C1)=O N1(C(C2(CC=C)CC2)=O)CC(NC(c2cc(C)c(C)o2)=O)CC(C)(C)C1 N1(C(C#C)(C)C)CCN(C(=O)C(=O)NCc2cccnc2Br)CC1 C=CCCCC(=O)NC(C1CN(C(=O)C(c2ccc(Cl)nc2)(C)C)CCO1)C C(=O)(CC(C)C(C)(C)C)NC(C)CC1CN(C(c2coc(C(F)F)n2)=O)C1 n1(CCC(=O)N(C)CC2CCN(C(=O)CCc3cnn(C)n3)C2)cnccc1=O N1(C(=O)C2=CCCCO2)CC(NC(C2(F)CC3(CCC3)C2)=O)C2CCCCC12 Cc1cc(Cl)c(C(=O)NCCC2CC(NC(=O)C(C)Cn3ccnc3)C2)cc1N C1(COC)CN(C(=O)C(c2ccccc2)=O)CCN1C(c1cccnn1)=O O=C1Cc2c(N(C3CC(N)C3)C(=O)Cc3cccc(Br)c3)ncnc2N1 CCCC(C(=O)NCC1CC(NC(=O)C(C)(C)CF)CCO1)S(N)(=O)=O CCCCCC(CC)C(=O)NC(C1CCN(c2cc(CCC)nc(Cl)n2)C1)C c1(C(=O)NCC(CNC(C(=O)NC(=O)NCC)C)O)ccc(Br)nc1N c1(C(N2CCCC2c2ccc(F)cc2)C(=O)NCCOC)cc(Cl)nn1C c1(C(N(C(C)C(N2CC(=O)NCC2C(C)C)=O)CC)=O)cc[nH]c2nccc1-2 C(CC(C)C)(C(=O)N(C)CC#N)N1CCN(c2cccc(OC)c2)CC1 c1(CCCCC(CNC(=O)OC)O)ccc(NCCC2(C)CC2(F)Cl)cc1 C(=O)(C1=C(Cl)CCC1)N(C(C1(CC2(OCC)CC2)CSC1)=O)C1CC1 C(C(CO)(CO)NC(=O)C=C1CCN(C)CC1)N(C(C(C)NC(N)=O)=O)C C(=O)(C1CCCc2cncn21)N1C(C)CN(C(c2cn(C(C)C)nn2)=O)C(C)C1 C(CS(=O)(=O)N(C)Cc1cnoc1-c1ccco1)(C1CCOC1)OC C1(N(C(=O)COCc2ccncc2)C)CCC(NC(c2nc(Cl)sc2Cl)=O)CC1 c1(N(C)C)nc(=NC(=O)NCC2COC3(CCC3)C2)[nH]s1 C(C(=O)NC(Cn1cccn1)C(=O)N(C)CCc1ncon1)(C(C)C)OCC N1(C(CC=CC=C)=O)CC(C)(C(=O)Nn2cncn2)CC1(C)C C1(C(N2CC(NC(C3CCC4(CC4)C3)=O)(CO)C2)=O)CCc2ncccc2C1 c1(CN(C(C2(F)CN(C(C=CC(=O)OCC)=O)C2)=O)C2CC2)cnccc1C Cc1ccc2c(c1F)N(Cc1cn(CCC(C)C)nn1)CCC2 N1(Cc2n(C)ncc2)CCc2[nH]nc(C(=O)Nc3c(Cl)ccnc3Cl)c2C1 C1(CCNC(c2c(C)occ2)=O)CSCCN1C(c1cccc(O)c1)=O c1(N2CCC3(CCN(Cc4cccc(OC)c4)C3)C2)c(F)cc([N+](=O)[O-])cc1F C12(CNC(C(C)c3ccon3)=O)CC1CN(C(=O)CCN1CCC1)C2 N1(C(c2cccc(NCC)c2)=O)CCCC2(CCC(NC(=O)C=NOC)C2)C1 N1(C(=O)C=Cc2ccsc2)CC2CCC1CC2NC(=O)C(F)(F)C1(O)CCC1 N1(C(CNC(CC(C)C)=O)=O)CCC2(CCN(S(=O)(=O)C(Cl)(Cl)Cl)C2)C1 C(CCN=[N+]=[N-])OCC(=O)NC1CC(CN(C(=O)CC2CCCO2)C)C1 c1(CC)nc(C(N2CCC2CC(=O)NC(C(O)CO)C2CC2)=O)c(C)o1 CC1C(=O)Nc2ccc(NC(C3CC4(CCC4)C3)=O)cc21 c1(SC)cccc(C(=O)NC(C)(CNC(=O)C(C)C(C)C)C2CCC2)c1Cl C1(c2nnc(CN(n3c(C)ncc3)CC3CC4CCC3C4)s2)CC2(CCC2)C(=O)O1 c1(CC(=O)NCC(C2CC2)NC(=O)CCCN2CCCC2)ccc(Cl)cc1 c1(COC)ccc(C(=O)NC2C(F)(F)C23CCC3)cc1C#N c1(C(N(C2CC2NC(=O)C=C(Cl)Cl)C)=O)ccc(N2CC=CC2)cc1 C1(CCNC(CC(CC=C)(C)C)=O)CCN(C(C2CCOC2C)=O)CCC1(F)F CC1(C)CC(NC(c2ccc([N+](=O)[O-])cn2)=O)CCN(C(C2COC(=O)N2)=O)C1 C1(C(=O)NC(C(c2ccccc2)NC(C(C)C)=O)C)Cc2cccc(F)c2O1 N1(C(CN(C(=O)C(F)C2CC2)C)=O)CCN(C(C2C=CCCC2)=O)CC1 C1(C(N2CC(NC(c3ccc(COC)o3)=O)C(OC)C2)=O)CCCC(C#N)C1 C1(NC(=O)C=CCF)CCCN(C(=O)Cc2ccnc(Cl)c2F)CC1 C(C#Cc1ccccc1)NCCN(CCC#N)CC Cc1[nH]c(C#N)cc1C(=O)NC1CCC(N(C(=O)Cc2cc(F)ccc2F)C)C1 C1(C)(CNC(C(COCC)n2cc(C3CCCC3O)nn2)=O)CC=CCC1 c1(-c2cn(CCN(C)C(c3c[nH]ccc3=O)=O)nn2)cccc([N+](=O)[O-])c1 c1(CC)noc(CN(CCNC(=O)CC(C)C2CCCO2)C2CC2)n1 n1(CC)cc(C(C)NC(=O)C(C2CC2)NC(=O)Cn2cc(C)nn2)cn1.C1CC1 C1(NC(c2cc(=N)[nH]cc2)=O)CC2CC1CN(C(=O)COCc1ccccn1)C2 CC1(C)CCCC(C)(NC(C2CCC3(CC3)N2C(=O)CC2=CCCC2)=O)C1 C(=O)(C1CCCc2ccnn21)NCC1(CO)CCCN(C(CC(C)F)=O)C1 C1(C(N(CCC(=O)NCC(C=C)(C)C)CCCO)=O)CCCC(C)CC1 C1(C(N(CCNC(COCCC#C)=O)C2CC2)=O)CC1C1CCCC1 CC1(C)CC(CC(=O)N(C2CCCC2)CCCNC(=O)CC2CC(F)(F)C2)C1 CCCCN=C(NCc1cnc(C2CC2)o1)NCC(c1ccccc1C)(C)C c1(CNC(CCC)(C)C)cc(C)cc(C)c1.C12CC1C(=O)N2 C(CCCCCC(=O)N(CC(C)C(=O)OC)C)NC(C(CC(=C)C)OC)=O c1(CNC(=O)C(N2CCCC(COCC3(C(F)F)CC3)C2)=O)cc(F)ccc1F Cc1cc(C)c2c(c1)C(N(C)C(c1ccc3c(c1O)CCCC3)=O)CCO2 C12(NC(C3C(C)C3C)=O)CC(CNC(c3n[nH]cc3Cl)=O)(C1)OC21CCC1 N1(C(c2cn(CCC)nn2)=O)CCC(O)C(NC(C2CC2C(C)(F)F)=O)C1 N1(C(CCCNC(N)=O)=O)CCOC(CCCCNC(C2CC3CC3C2)=O)C1 N1(C(C(C)(C)OC)=O)CC2CCC2(C(N2CC3CC2CN3C(C)=O)=O)C1 S(=O)(=O)(c1ccc(Br)cc1NCC1CC(OC)C1(C)C)NCCNC(=O)NC C1(C(=O)NC2CN(C(COCC(=C)C)=O)CC(F)C2)CC(c2cnn(C)c2)=NO1 c1(N2CCN(C(c3c(OC)ccc(OC)c3)=O)CC2)cc2c(cn1)C(=O)CCC2 c1(C(=O)NCC23C(CN(C(CCOC)=O)C2)C3)ccc(C)c(Br)c1C C(=O)(NNC(=O)c1cc(Br)ccc1)c1cn(C(C)(C)C)nn1 c1(Cn2ncc(C(C(=O)NC3CCC3)N(C(C)CC#N)C)c2)ccc(Br)cc1 c1(OC)ccc2[nH]cc(C(N3CCN(Cc4cnc(F)cc4C)C4CC34)=O)c2n1 C(CC(=O)NC(c1nccs1)C1CCC1)(C1CCCCC1)OC(=O)NC(C)(C)C c12ccc(cc1)C(=O)NC2CN(C)C.n1(CC#C)ccc(NC(=O)C=CCC)c1 c1(C(=O)NCCCN(C(c2ccc(F)c(CO)c2)=O)CC)cc(F)c(F)cc1O N1(Cc2nn(CC)nc2C)CCC2(CCN(C(C3CC3c3ccccc3)=O)C2)C1 O=C(C1=CCCOCC1)NC(CNC(C1CCCCCS1(=O)=O)=O)CC(F)(F)F Cc1cc(C)c(CC(=O)NC2CCC(O)CN(C(=O)Cc3cc[nH]c3)C2)c(O)n1 C1(NC(CC(=O)OCC)=O)CN(C(=O)CC2CCCN2C)CCC1(F)F C1(NC(COCC(=O)OC)=O)CCCC(C(=O)NC(C2CN(CC(C)C)C2)=O)C1 c1(CC)ccc(C(=O)NC(CNC(C2COC(=O)N2C)=O)CC(C)C)nc1 N1(C(c2cncc(NC)c2)=O)CC(CNC(=O)Cc2cscc2F)C2(CC2)C1 CCC(C)(CC)C(=O)NCCC1CCCN1C(=O)C(=O)Nc1ccc(Cl)c(F)c1 C1(NC(=O)CC2CC2)CN(C(c2nc[nH]c3nccc2-3)=O)C2(CCCC2)C1 c1(C(N(C2CCN(C(c3coc(Cl)n3)=O)C2)CC)=O)nnccc1C c1(NC(c2n(CC)ncn2)=O)cccc(NC(=O)CCC2CC(C)(C)CO2)c1 n1(C(C)(C)C)nnnc1C(C)(CCN1CCSCC1)NCCC1CCOC1 C1(O)(CNC(c2cc(CNC(C(C)(C)SC)=O)[nH]n2)=O)CC2CCC1C2 Cn1nnc2c1C(C(=O)N1CC3(C1)CN(C(C1CCC1)=O)C3)CCC2 C(=O)(CC(C)CCC=C(C)C)N1CC(COC)N(C(=O)CC2CC3(CC3)C2)CC1 c1(C(=O)NC2C(CNC(c3cn(CC)nn3)=O)CCC2)c(C)ccc(Cl)c1F C1(CCNC(CSC(C)C)=O)CCC(NC(c2csc(C(C)C)n2)=O)C1 C1(C(=O)NC(C)CNC(=O)C(C)(C)N2CCCCC2)CCCCC12CCC2 c12cc(ccc1C)COC2=O.C1(NC(C2C(C(=O)OC)C2)=O)CN(C(C)C)C1 c1(CC(=O)NCCOC(CNC(CC(C)C2CC2)=O)(C)C)nc2ncccn2n1 C1(NC(C2(CC)CCC2)=O)CN(C(c2csc(N(C)C)n2)=O)CC1CNC(C)=O C1(CCNC(c2cnn(C(F)F)c2)=O)CN(C(c2cnnn2C2CC2)=O)CCO1 C1(NC(CCCC2(C)N=N2)=O)(CF)CCN(C(=O)C(c2ccc(C)cc2)O)C1 c1(C(CC)=O)ccc(C(=O)NCC2CCC(NC(C3CC4(CSC4)C3)=O)C2)cc1 c1(C(=O)NC2(CC(=O)Nc3cc(C#N)ncc3)CCC2)cccc2c(Br)n[nH]c12 C(=O)(C(C)(CNC(=O)CC1OCCO1)CC)NC1(C#C)CCOC1 Cc1ccc(NC(=O)CNC(C2CCCN(C(=O)C(F)n3cccn3)C2)C)cc1 C1(CC2(C)CC(OCc3ccccc3)C2)CCCCC12CC2(F)F C1(NC(c2cc(C)ns2)=O)C2CC(O)C1N(C(=O)CNC(C1CCOCC1)=O)C2 C12CCC(CC1)NC(=O)c1scc(n1)C(=O)N2.c1(CC2CC23CC3)ccccc1 CC(C)(O)C(F)CNC(=O)C(CCC1CC1)NC(=O)C(=O)NCC(F)F N1(C(=O)CCF)CC2OC(=O)N(C3CCN(C(=O)COCC4CC4)C3)C2C1 C1(C(=O)NCCOCCN2CCOCC2)CCC(n2cc(C(O)C3CC3)nn2)CC1 C(=O)(C1Cc2ccc(Cl)cc21)NCC(CNC(c1nccc(OC)c1)=O)OC C1(CC(=O)NC2(CCNC(C=CCCC)=O)CCC2)CC2(CCO1)CC2 C1(C(N(C2CCN(C)CC2)C)=O)CCN(C(=O)CC2CCCC(=O)C2)CCO1 N1(C(c2c(CNC(C(CC#C)O)=O)ocn2)=O)CCC(O)C(F)C1 C(=O)(CCCS(N)(=O)=O)NCC(CN(C)Cc1n[nH]c(C2CC2)n1)O c1(C(N2CCC(NC(C3=C(C)OCCS3)=O)C(O)C2)=O)cccc2ccn(C)c12 C(CC)(C(=O)NCCC1CCC(NC(=O)C(CC)Oc2ccccc2)C1)=CC c1(OC)c(C(N2CCC(C)(NC(=O)CSC(C)C)C2)=O)cc(Cl)cc1Cl c1(C(N2CCC(O)(C(CNC(C3(C)CC(=C)C3)=O)C)C2)=O)cc(C)ccc1Cl Cn1ncc2c(NC(=O)NC3CCCCCC3(F)F)ccnc12 N1(C(CC(C2CCCCCC2)N)=O)CCSC(C(F)(F)F)C1 c1(NC2CN(C(CCCN(C(C)=O)C)=O)CC2C)ncc(Br)cc1[N+](=O)[O-] C12(NC(c3cnc(OC)s3)=O)CCC(CN(C(=O)Cc3ccsc3)C1)C2 O=S(=O)(c1ccc(NCc2cc(O)ncn2)c(F)c1)NCc1ncccc1Cl C(CCCC(=O)NCC(CNC(C1COC(=O)O1)=O)CO)N(C)C c1(C(=O)NCC2CN(C(C3N(CCCC)CCCC3)=O)C2)cc(C)nc(O)n1 C1(NC(C(C)NS(CC)(=O)=O)=O)(CNC(c2cccnc2F)=O)CCCCC1C Cc1[nH]cc(C(N2CC=CC2CNC(c2cnn(C)c2Cl)=O)=O)c(=O)c1Cl C1(C(=O)NC2CN(C(C3(CC(C)C)CCC3)=O)CC23CC3)CC2CCC(C1)C2=O C=C(Cl)C(C)(C)C(=O)NCC1(NC(c2cc(CO)c(C)o2)=O)CCOC1 c1(OC)cc(F)c(C(=O)NCC2C3CN(C(=O)Cc4nncn4C)CC23)cc1N CC(C1CCCCC1)=CC(=O)NC1CC2CCC1N2C(=O)C(C)(C)C(N)=O N1(C(C(CCC)NC(=O)COC)=O)CC(=O)NCC1c1ccccc1 C1(CC)CCCCC1C(=O)N(CCNC(C1CCCN(C(C)=O)C1)=O)CCOC C(CC(CNC(=O)C(C)CSCc1ccccc1)NC(c1cc(C)[nH]n1)=O)OC S(=O)(=O)(c1ccc(NC2CCC2O)c(Cl)c1)NCc1c(F)ccc(C)c1F C(=O)(C1=CCCSC1)N(CCCC(=O)NC1C(OC)CCCC1)C C1(C(=O)NC2(COC)CN(C(C3(C)CCCS3)=O)C2)CCc2nnnn2C1 C(=O)(C1CCc2cc(F)ccc21)NC1(CCOC)CCN(C(C2CSC2)=O)C1 C1(C2(O)CCN(C(=O)C3=CCOC3)CC2)(NC(C2CCC(C)C(C)C2)=O)CC1 C1(CC(=O)NCCCCCC)CN(C(=O)CCCSC)C(C)(C)C1 c12ccc(c(OC)c1)OC(=O)C1CCN(C1)C2=O.C(C(=O)N(C1CC1)CC)CC N1(C(C(N2CCOC2=O)C)=O)CCOC(C(N2CC(n3ccnc3)C2)=O)C1 N1(C(CSCC#C)=O)CCCCC1C1CCCN1C(=O)CCc1nc(C)cs1 C1(O)(C(C)NC(C(C2CC2)OCC)=O)CCN(C(c2c(C)nn(C)c2Cl)=O)CC1 n1(CC(=O)NC2(CF)CCN(C(C(C)C#N)=O)C2)cc2ncccc2n1 c1(C(N2CCC(CO)C2)=O)cc2cc(-c3cnn4cccnc34)ccn2n1 C1(CNC(C(C(C)C)n2ncc(C)c2)=O)CN(C(=O)CC2CSC2)CC1(F)F C(=O)(C(C)CCC(C)(C)C)N1CC(CN(C(=O)C=CCn2cncn2)C)OCC1 c1(CC(=O)NC(C(=O)N(C(C=C)C2CC2)C)CC2CCC2)cccnc1F C1(C(=O)NCCCCCOC)CN(C(=O)C(c2ccn(C)n2)C)C2(CCC2)C1 c1(CC)cc(C)c(C(=O)NC2CC3(C2)CC3NC(c2ccc(SC)o2)=O)o1 C1(NC(CC2(OCC)CC2)=O)CCN(C(c2ccco2)=O)CC(C)(C)C1 c1(C(=O)NCC#CCNC(=O)C2=C(Cl)CCOC2)cnc2ncnc(O)c2c1 C(=O)(CCCCCCNC(=O)CC1CC(N(C)C)C1)N(CCC(=O)OC)CC CC1CC(NC(c2ccc(C3CC3)cc2)=O)CN(C(c2cc(F)ccc2O)=O)C1 c1(C(=O)NCCC2CCN(C(c3csnn3)=O)C2)ccc2c(F)cc(F)cc2n1 N1(C(c2cn(C)nc2C2CCOC2)=O)CC2CCCN(C(=O)CC3CCC3)C2C1 c1(C(N2CC3CC(CNC(CCCC(N)=O)=O)C3C2)=O)ccnc2ccc(N)cc12 CC1(C)CC(C)(C(=O)NCC(C2CCCC2)NC(c2ccn(C3CC3)n2)=O)C1 c1(OC)cc(C(=O)NCC(C(C)C)NC(=O)COCCCN=[N+]=[N-])ccc1F Cc1ccc2[nH]cc(CNC3CN(c4ncc(C)cn4)CC3C)c2c1 C1(C(=O)NC(C(=O)N(C(C)CC(F)(F)F)C)C2(O)CCC2)CCCC2(CC2)C1 C1(C(=O)NCC2N(C(CCNC(C)=O)=O)CC(O)C2)CCCC1C1CC1 N1(CC2CCN(C(=O)CCC(F)(F)F)CC2)C2CCC1CC(NC(C1CCO1)=O)C2 CN1CCC(n2cc(NC(N3CCCC3c3nc(N(C)C)no3)=O)cn2)CC1 c1(CNC(CN2CCC(O)(c3n(C)ncc3)CC2)=O)cc2c(cc1Cl)OCCC2 C1(CNC(C(C(C)C)C2CCC2)=O)CN(C(=O)CCCC#N)C2CCN1C2 C(=O)(C(C(C)C)N1CCCCC1)NC(CC)CNC(=O)Cn1cc(Cl)cn1 c1(C(=O)NCC2C(NC(CC3CCC(=O)O3)=O)C2)cnc2ccccc2n1 N1(C(CC(C=C)CCC)=O)Cc2ccccc2C(NC(=O)CN2CC3CC3C2)C1 c1(C(=O)NCCN(C(C(C(C)OC)O)=O)C2CCCC2)cc2c(cn1)CCCC2 N1(C(C2(CC=C)CC2)=O)CC(C(C)(C)O)(CNC(c2cnc(Cl)s2)=O)C1 O=C1NCCCCC1C(N1CCC(CCCNC(=O)C(F)(F)C(F)F)CC1)=O N1(CCONC(=O)C2(CC(=O)NC(C3CCCO3)C)CC2)CCCC1 C1(CCNC(CSCC=C)=O)CN(C(C)=O)CCO1.c12ccc(o1)CNC2=O Cc1c(C(=O)Nc2ccc(NC(C3(CC#N)COC3)=O)cc2)cccc1CO Cc1c(C(=O)N(C2CCN(C(=O)C=Cc3cnc[nH]3)C2)C)oc2c(C)cccc12 C1(C(N2CCC(N(C(c3c(C)scn3)=O)C)C2)=O)CCC(C)CC1 CC1(C)CN(C(C2CCCCN2C(c2csc(O)n2)=O)=O)CC1O N1(C(c2c(C)n[nH]c2C)=O)CC(NC(c2ccc(Cl)cc2)=O)CC(O)C1 C1(NC(C2CCC(C)O2)=O)C2CC3C(C2)C13C(=O)NC1CCN(C(C)(C)C)C1 n1(CCC=C)cc(C(=O)NC2(C3CCCN3C(=O)CNC(=O)CC)CC2)cn1 C1(CN(C(C2SC3C=CC2C3)=O)CC)CCN(C(=O)C=CC(=O)N(C)C)CC1 CC1=C(C(=O)NCC(O)CNC(c2c(C)noc2-c2ccccc2)=O)CCCC1 c1(N2CC(O)(CNC(C3C(C)CC(=O)N3)=O)C2)cc(=O)n(C)c(=O)n1C c1(C(N)=O)cccc(NC(C2CC2NCc2csc(Br)c2)=O)c1Cl C(=O)(C1CCCc2c[nH]nc21)N1C2C(NC(c3cncc(Br)c3)=O)C(C2)C1 c1(OCC)cc(N2CCC(N(C(=O)CC3C=CCCC3)CC)C2)ccc1[N+](=O)[O-] Cc1cc(-c2nc(CC3CC3)nn2-c2cnnn2C)c2ccccc2n1 Cc1ccc(C(=O)NCC(C)NC(=O)CCC2CCCO2)cc1[N+](=O)[O-] C1(CC(=O)NCC2(F)CC(CNC(c3ccsn3)=O)C2)(COC)CCCC1 C1(C)(OC)CCCN(C(=O)C2=CCN(C(=O)Cc3csc(C)n3)C2)CC1 c1(C(N2CCC(CNC(CCCCC)=O)(OC)C2)=O)cc(C)c2nc(C)cn2n1 N1(C(CN(CC)CC)=O)CC(NC(=O)CC2C=NN(C)C2=O)CC1(C)C CC1CC(NCc2ccc(C#N)cc2)CC(C)(C)C1 N1(C(C2N(C(CC)=O)CSC2)=O)CC(CN(C(=O)C(F)(F)CC)CC)C(C)C1 Cc1cc(Cl)cc(Br)c1NC(c1nc(C(=O)OCc2c(F)cccc2F)sc1)=O c1(CN(C(C2CC(C)C2)C(=O)NCc2nnn(C)n2)C)c(Cl)cccc1Cl N(C1CCCn2cnnc21)C(C(CC1CCC1)NC(COCCOCC)=O)=O c1(C(C(=O)NCCCCCCNC(=O)CC2CCC2)O)ccc(Cl)cc1Cl CS(=O)(=O)c1cnc2c(C(=O)Nc3ccc4c(O)n[nH]c4c3)cnn2c1 C1(NC(C(C)N2CCC2)=O)CC(F)CN(C(c2ccc(C(F)(F)F)cc2Cl)=O)C1 c1(N2CCC(C(C)NC(=O)CC3CCCOC3)CC2)ccc(C#N)cc1[N+](=O)[O-] C1(NC(C2(CCOC)CC2)=O)CCN(CCNC23CC(C(C)(F)F)(C2)C3)CC1 C1(NC(C(CC)(C)CO)=O)CC2CCC1CC2NC(=O)CC1CNC(=O)O1 N1(C(C2(CNC(=O)CC(=O)NCC)CC(=C)C2)=O)CCC12CCCSC2 N1(C(CNS(C)(=O)=O)=O)CCC(NC(=O)CCOCC2CCCO2)CC(O)C1 C(C(=O)NC1CN(C(=O)C=CC(F)(F)F)CC(C)(C)C1)(c1ccccc1)=C(C)C N1(C(C2CCSC2)=O)CCOC(C(=O)NCCCNC(c2ncccc2O)=O)C1 Cc1nc(C(=O)NC2(CNC(c3ncc(Cl)cc3F)=O)CCC2)cn(C)c1=O N1(CCOC)CC(C(N2CCOC(CNC(C3(O)CCCCC3)=O)C2)=O)CC1=O C(c1ccnn1C)=CC(=O)NCC(CC=C)NC(=O)C(O)CCN(C)C c1(N2CC(CNC(=O)CCc3cccnc3)OCCC2)ncnc2cnccc12 c1(C2CCN(c3n(CCC#C)c(-c4cnc(C)[nH]4)nn3)C2)ccc2c(c1)OCO2 CCCCC(C(=O)NC1(C)CCCCC1C)NCC12CCN(CC1)C2 N1(C(Cc2ccc(OC)c(O)c2)=O)CCC2C1CCCN2c1ncncc1C#N c1(C(N2CC(NC(C3C(C=C)C3)=O)C2)=O)cn(C)nc1-c1ccco1 C(C(CC(=O)N1CC(CNC(C2(N(C)C)CCC2)=O)C1)C(F)(F)F)N(C)C C(C(CC(F)(F)F)NC(c1ccc(OC)s1)=O)NC(c1cc(CC)on1)=O c1(C(N2CCOC(c3nc[nH]n3)C2)C(=O)NCCC)cccc2[nH]ncc12 C1(NC(CC2C(C)CCC2)=O)CCC(NC(c2nccc(C(F)F)n2)=O)CC1 N1(C(CCOCCCNC(c2ccc([N+](=O)[O-])o2)=O)=O)CCOC2C(O)CC12 c1(CC)ccc(C)c(C(=O)NC(C)C(C)(C)NC(=O)C(F)CN(CC)CC)c1 C1(NC(C)=O)CCCN(C(=O)NCc2c(OC(F)(F)F)cnnc2OC)CC1F C1(C(=O)NCC2(C)N(C(CCC3(C)N=N3)=O)CCC2)C2CCC(C2)C1(C)C c1(C(=O)NC2CC(NC(C3CC(OCC)C3)=O)C2)cc2cc(Cl)ccc2o1 CCCC(C(O)C(=O)NC(C(=O)NC)C1CC1)NC(=O)C(c1ccccc1)O CCC(C)C(O)C(C)C(=O)N1CC(C(O)C(=O)NC2CCOC2(C)C)C1 Cc1coc(C2CC2)c1C(N1CCC(C)(CNC(c2cc(Cl)cnn2)=O)C1)=O C(=O)(C1=CCCN(C(=O)CC(=O)OC(C)(C)C)C1)N1CCC(N(C)C)CC1 C(=O)(C1=CCN(C(c2ncnc(O)c2F)=O)CC1)NCC(c1nccs1)C N1(C(Cc2nc(C)sc2)=O)CCC(F)(CNC(c2sc(O)nc2C)=O)C1 c1(N2CC=CC2)nc2c(c(=NCC3CC4C(C3)C4(F)F)[nH]1)CCCCC2 N1(C(CC2(C)CC2(F)F)=O)CCCC(NC(c2ncccc2N)=O)CC1 N1(C(CCc2cnc(C)o2)=O)CCC(C(CO)NC(C2CCC(C)(C)C2)=O)CC1 c1(OC)ccc(C(=O)N(C2CN(C(=O)CCc3nc(C)no3)C2)C)c(F)n1 CCCC(CC)CC(=O)NC1CC(NC(=O)C(c2ccccc2Cl)(C)C)CC1O c1(CC)c(Cl)nc[nH]c1=NCc1ccc(C2CC2)cc1F c1(CN(C2CCN(C(Cn3nnc(C)n3)=O)C2)C)cc(F)c(F)c(Cl)c1F N1(C(C=C2CCC(C)C2)=O)CCC2(CCCN2C(=O)CCC(=O)C2CC2)CC1 N1(C(CC=C)=O)CCCC(O)(CNC(=O)C(C)(C)S(C)(=O)=O)CC1 c1(C(N2C(CCNC(c3conc3C(F)(F)F)=O)CCC2)=O)n[nH]c2c1COC2 Cc1cccc(CC(=O)NCCC(C)N(C(=O)CC2CC3(CC3)CO2)C)c1F N1(C(c2cc(OC)no2)=O)CCOCC1CNC(c1sccc1Br)=O C(c1ccc2c(c1)OCO2)=CC(=O)N(C)CC1CCN(C(C(CCCC)O)=O)C1 N1(C(CC(C)CF)=O)CCN(C(C2(c3cccc(F)c3)CCC2)=O)CC2(CC2)C1 Cc1c(C(=O)NCC23CC(NC(=O)COCC(C)C)(C2)C3)cccc1C(F)(F)F C(C)(CNC(=O)C(c1ccn(C)n1)C)(CNC(=O)C(C)(C)n1cncn1)OC Cc1nn(C)c2c(NC(c3ccc(Cl)cc3F)C)nc(=NC3CCCOC3)[nH]c12 c1(C(C)NC(=O)Nc2cccc(Br)c2Cl)nc2c(o1)CCSC2 CC(C)C(N=c1nc[nH]n2cccc12)C(C)NC(c1ccnc2ccsc12)=O c1(C(C)=O)cccc2ccc(C(=O)COC(=O)Cn3nnnc3C)nc12 CC(C)CC(O)C(C)C(=O)NCC(O)CNC(C1(N(C)C)CCCCC1)=O C(CCF)(C(=O)N1CC(F)(C#N)C1)NC(Cc1nc(C)oc1)=O Cc1nnc2n1CC(C(N1CCC3(C1)CN(C(=O)COCP(C)(C)=O)C3)=O)C2 N1(C(C(CC2CC2)OC)=O)CCC(CNC(c2n[nH]c3c2COC3)=O)C(F)(F)C1 CC1(C)CC(C(=O)NCC2(n3cnnn3)CC2)CN1C(=O)CC1CC=CCC1 C1(NC(c2ccc(N(C)C)nc2)=O)C2CC3CN(C(C4C5COCC45)=O)C1C3C2 N1(C(c2c(CC)c(C)sc2)=O)CC2CCC(C1)N2C(=O)COC1CCCCC1C C1(CC)CCN(C(=O)CC2(C#N)CC2)C(C(=O)NC23CCC(CC2)C3)C1 c1(C(=O)NCC2(N)CC2)ccncc1Nc1ccnc(Br)n1 Cc1cn(C)nc1C(=O)NCC1CN(C(=O)CC(O)Cc2ccccc2)CC1O Cc1cc(Cl)cc(C(N2CC(NC(=O)CN(C)C(=O)C3CC3)CC(F)C2)=O)c1C N1(C(C(C)OCC=C)=O)CCC(NC(C2(CC)CCOCC2)=O)C1C1CC1 N1(C(C2(SC)CCC2)=O)CCC2(CCCC2CNC(=O)CC2CC2C)CC1 CC1=NNC(=O)C1CCC(N1CC(NC(C2(NC(C)=O)CCCC2)=O)C(C)C1)=O C1(C(=O)NC(c2nc(C)[nH]n2)(C)C)CN2CCN1CC2C c1(C(c2nnnn2C2COC2)NCCn2c(=O)ccnc2)ccc(Br)cn1 c1(C(N2CCN(C(C3(C)CCNC3=O)=O)CC2CO)=O)cc(Cl)cc2c1OCC2 C1(NC(c2c(CCC)[nH]cc2)=O)CCN(C(=O)COc2ccc(Cl)nc2)CC1C CC1C(NC(=O)CCOC2CC2)CCCN1C(c1cc(CCO)on1)=O Cc1ccc(C(=O)NC2CS(=O)(=O)CC2NC(c2cccc(C)c2C)=O)c(F)c1 Cc1noc(C)c1-c1cn(CC2CCCN2C(C2CC3CCCC23)=O)nn1 N1(C(c2n[nH]c(C)c2Cl)=O)CCC2(CC1)CC2CNC(C1CC(=C2CCC2)C1)=O Cc1c(C(N2CC(CC3CCCCN3C)C2)=O)nnn1CCn1cc(CO)nn1 N1(C(C(CC=C)(F)F)=O)CCC(C(=O)NCCC2(O)CCC2)C(C)(C)C1 C(CNC(=O)C(C)(C)C1CCOC1)(CC(=O)NC(c1cnsc1)C)OC Cn1c(=O)c(SCCC(C)(C)O)nc2ccccc12 C1(C(=O)NCC(C(C)C)(C)NC(c2cc(C3CC3)no2)=O)Cc2nncn2C1 CCCCC(CNC(=O)CSc1nnc(C)n1C)NC(=O)COCCC c1(C(=O)NC(CC=C)CNC(c2cc(O)cc(O)n2)=O)cc(C)c(C)cc1C N1(C(=O)Cc2cccc(OCC(F)(F)F)c2)CCN(C(=O)CC(F)F)C(CO)C1 C1(O)(CCNC(CCc2cccc(OCC)c2)=O)CCCN(C(C2(O)CC2)=O)C1 c1(OC)c(F)ccc(F)c1CN1CCC(NC(=O)CCc2ncc[nH]2)C(O)C1 Cc1ncc(C=CC(=O)N(C(C)CNC(=O)CC2CCN(C)C2=O)C)c(O)n1 C(=O)(C1CCCc2n[nH]cc21)N1CC(COC)(CNC(c2cccc(SC)c2)=O)C1 N1(C(C2N(C(c3nc(C(C)C)oc3)=O)CC=C2)=O)CCC2CC1C(=O)O2 C1(CNC(c2c(C)onc2)=O)CC2CCC1N(C(=O)C(C)C(C)(F)F)C2 C1(N(C(C2(CNC(CCC3CC(OC)C3)=O)CCCO2)=O)C)CC2CCC1O2 N1(C(c2ccc(CC)[nH]2)=O)CCN(C(c2cnn(-c3nccs3)c2)=O)CCC1C N1(C(C(C(=O)OC)C)=O)CCC(O)(c2cn(CCCCCCF)nn2)CC1 Cc1c(C(=O)NC2CN(C(c3ccsc3C#N)=O)CC2C)oc2c(C)cccc12 c1(C(=O)OCC2CCC3(C(C(=O)OC)C3)C2)ccc2oc(=N)[nH]c2c1 CC(C(=O)NC(c1nocc1C(=O)N(C)CCc1ccccn1)C)C(C)(C)C C12(C(=O)NCC3C4CN(C(C(=O)NCCCC)=O)CC43)CCC(OCCC)C1CC2 C1(CNC(C(N2CCN(CCC(C)C)CC2)C(C)C)=O)Cc2cc(Br)ccc2O1 C1(N(C(C=Cc2ncc(C)[nH]2)=O)C)CN(C(=O)CCC2CCC2)CC1(C)C O(NC(=O)C(CCF)NC(=O)C(F)CCCCC)CCOCC#C C1(OCCC)CN(C(=O)C2CC2)CC1CNC(C1(O)CN(CC)C1)=O N1(C(CC(CN(C)C)C(F)F)=O)CCC2CN(C(=O)C(C)(Cl)Cl)CC2C1 C1(N(C(CCN(CC)CC)=O)C)CCCC(NC(=O)C=Cc2ccncc2)C1 C1(N(C)C(C2CCC3CC3C2)=O)CC2CCC(C1)N2C(c1ccncc1O)=O Clc1cc(NC(c2sccc2Cl)c2nnnn2C2CCOC2)cc(Cl)c1 c1cc(=NC2CC3(CCCO3)C2)[nH]c(N2CCOC(C3CC3)CC2)n1 C1(OC)CN(C)C(C)(C(N2CC(CNC(c3cn4c(n3)SCC4)=O)C2)=O)C1 CON(CCC(=O)N(CC(O)C(F)(F)F)C)C(=O)C(F)C1CCOCC1 C1(C(=O)NCCSC(CC)C)(NC(=O)C(C2CCC2)N(C)C)CCC1 N1(C(CCC(C)C)=O)CC2(C1)CN(C(C1CCOC1)=O)C2.C1C(=O)N1 c12cn(C)nc1NC2=O.c1(CCNC(CN(CC)CC)=O)ocnc1C.C(C(F)F)O C1(C(=O)NC2(CC(=O)OC)CC2)(NCCC2CCCO2)CC(O)C1 c1(OC)c(Cl)nc[nH]c1=NCC(C)(C)C1CN(C(C2CCC(=O)N2)=O)C1 c1(OC)cccc2c(N3CC4CC3C3CC43)cc(C)nc12 C1(O)(CNC(CN2CC(C)(C)C2)=O)CCCN(C(C23CC2COC3(C)C)=O)C1 N1(C(c2cnc(C(C)C)o2)=O)CC(NC(=O)C=CC2CCOC2)C(C)C1 C1(NC(C(CCC)OC)=O)CN(C(=O)CSCCC(C)C)C2CCCCC12 N1(C(CCNC(=O)NC)=O)CC(CO)C2(C1)CN(C(C1CN(C(C)C)C1)=O)C2 c1(OC)ccc(C=CC(=O)NC(C)CN(C(=O)C(C)NS(C)(=O)=O)C)c(C)c1 C1(C(=O)NCc2n(CC)c(C)nc2)CCN(C(=O)CN2CCOC2=O)O1 n1(C(C(=O)NC2(CNC(CC=CC=C)=O)CC2)C)ccc(C)n1 C1(CNC(c2n(CCC)nnn2)c2cc(C3CC3)ns2)CC(F)(F)CO1 C1(C(N2CCC(NC(c3c(C#C)c[nH]n3)=O)(CF)C2)=O)CCc2ncc(C)n2C1 C1(CNC(CSC(C)(C)C)=O)CCN(C(=O)CC2COCCO2)CC1(F)F C(N=c1[nH]c(C(F)F)nc(=N)[nH]1)C1N(C(CC2(NC(C)=O)CC2)=O)CCCC1C N1(C(CCNC(C)=O)=O)CCCC(F)(CNC(C2CCNC(=O)C2)=O)C1 C(=O)(C(F)(CNC(c1ccc(C)c(C)n1)=O)C(C)C)NC1(CSC)CCCC1 Cc1cc(C(N2CC3CC2(CNC(=O)CC(C)n2cccn2)C3)=O)ccc1N c1(C(=O)NC2CC(C(=O)NC(C=C)C)C2)ccc(OC(C)C)cn1 c1(CCNC(N(CC(C2CCC2)OCC)C)=O)ccc(F)cn1 c1(CN(C)C)n[nH]cc1C(=O)NC1CC1NC(C1(C)CC1(C)C)=O N1(C(CN(C)C(C2CC2F)=O)=O)CCN(C(c2c[nH]nc2Br)=O)CC1 N1(C(CC=C)=O)CC2CC2(CNC(c2cn(CC3CCOCC3)nn2)=O)C1 C1(c2n(C(C)C)nnn2)(NCCNC(=O)OC(C)(C)C)CC2(C1)CC(C)(C#N)C2 C1(CNC(c2cnc(Cl)c(Cl)c2)=O)CC2CCC1N(C(=O)COCC(F)F)C2 c1(C(N(C2CCN(C(C(C)c3cncs3)=O)C2)C)=O)cccc2cncn12 C1(NC(C(N2CCOC2=O)C)=O)CC=C(C(=O)NCc2cccc(O)n2)C1 C(=O)(CCCCCC#N)NC(CCOC)CNC(=O)C1CC1 C1(Cl)(C(=O)NC(c2ccc(CC(C)C)cc2)C)CC2CCC1O2 c1(C(=O)NC2CCN(C(CC3(OC)CCCC3)=O)C2C2CC2)cc(O)nc(O)c1 C=Cc1ccc2c(c1)CN(C(=O)C(n1c(=O)n(C)c(=O)c3ccccc13)C)C2 c1(C(C(=O)NCCSC)N(CCCC)CCCC)ccc(C)cc1Cl CC1(CNC(C2(OC)CC2)=O)CC(NC(=O)CCCNC(N)=O)C1.c1ccoc1 Cc1cc(C#N)cnc1C(N1CCCC1Cn1cc(Cn2ccsc2=O)nn1)=O N1(C(c2ccn(CCOC)n2)=O)CC2(CNC(=O)CC(C)(C)N(C)C)CC1CO2 c1(C(N2CC3C(CNC(C4CC4F)=O)(CC3)C2)=O)cc2cc(Cl)cnc2[nH]1 C1(C(=O)NCC(CC)(C)NC(c2c[nH]ccc2=O)=O)CCC2(CCC2)O1 CCCC(CC)CCC(=O)NCCCCNC(C1CCCCN1CC)=O N1(C(C2(CC=C)CCOC2)=O)CCC2(C1)CN(C(C13CC(F)C1C3)=O)C2 n1(CCC(=O)NC(CC(C)NC(C=CSC)=O)C)c(O)nc2ccccc2c1=O c1(C(N2CC(CC=C)(NC(=O)C(C)NC(c3cccs3)=O)C2)=O)cc(O)nc(O)c1 N1(C(C2ON=C(C)C2)=O)CCC(CC(N2CC(CC3CC3)C2)=O)CC1 N1(C(C(CCCNC(CCCC(C)(C)C)=O)O)=O)CC2(CCCCCC2)C1 CCC(C)(C)CC(=O)NC1CN(C(c2ccnnc2S)=O)CCC1c1ccccc1 CC1(C(N2CC3CC2CN3C(c2coc3c2CSC3)=O)=O)Cc2ccccc2N1 Nc1cc2c(cc1C(N1CCCC(CNC(=O)CC3CCSCC3)C1)=O)CCC2 CCN(C1CCCOC1)N1CCCC(NC(c2ccc(Br)cc2)=O)C1 N1(C(CCN(CCC)C)=O)CCCC(NC(C2CC3CC2CO3)=O)CC1 C1(NC(C(C)SC)=O)(CNC(=O)CCC=C(C)C)CCOC1 CC1(C)CC(NC(=O)CC2CCCC23CC3)CN1C(=O)CC(=O)NC1CC1 N1(C(c2nc(C)n(C)c2)=O)CCC(NC(c2cccnn2)=O)C(CO)C1 c1(C(=O)OCC)[nH]c(C)c(C(=O)NCCN(C(C2CCC(C)C2)=O)C(C)C)c1C N1(C(c2ccn(C)n2)=O)CCCC(C(=O)NC2CC2(C)C(F)F)C1 C(=O)(C1=NNC(=O)CC1)NC(CC)(C)CNC(c1cc(C)c(C)[nH]1)=O C1(NC(=O)CC2CC2)CC(O)CN(C(=O)CC2CC2C(F)(F)F)C1 c1(C(N2CC(C(=O)NCCNC(C(CSC)C)=O)C2)=O)[nH]c(O)nc1C C1(C(=O)NC(C2CCN(C(=O)C(C)(C)N3CCCC3)C2)C)CCc2n[nH]cc2C1 C12(NC(c3n(CCC)ccc3)=O)CCC(CNC(C3CC34CCC4)=O)(C1)OC2 N1(C(CC2CCC(C)CO2)=O)CC=C(C(=O)NCC(C)(CO)CO)CC1 c1(SCCC(=O)NC(C2(O)CCN(C(c3cncs3)=O)C2)C)ccc(F)c(F)c1 O=C(C(O)CF)NC1CCC1C(F)(F)F.c12cc(on1)CNC2=O N1(C(=O)OC(C)(C)C)CCC2C(C(=O)NC3CCN(c4ccc(Cl)cc4)C3=O)C12 CC1(C(=O)NCCOC2CCN(C(=O)CC3CCCO3)C2)CCCCNC1=O C1(C(C)C)CCC(C(N2CC(N3CCN(C(C4CC4(F)F)=O)CC3)C2)=O)C(=O)N1 C(C(F)(F)C(=O)N1CC(NC(c2ccnn2C2CCC2)=O)C(C(F)(F)F)C1)OC C(=O)(CC(C)C(C)(C)NC(c1ccc(O)nn1)=O)NC(c1cnn[nH]1)C N1(Cc2n(C(C)(C)C)ncc2)CCCC(c2cccs2)C1 C1(NC(C2Cn3c(C)nnc3C2)=O)CC2CCC1CN(C(=O)CC1=CCCC1)C2 N1(C(COCCCN=[N+]=[N-])=O)CCC2(CCCN(C(c3csc4nccn34)=O)C2)C1 C(CC(=O)N=c1ccn(C2CN(Cc3nc(C)ccc3C)C2)[nH]1)c1cnc(C)s1 c1(NCC2CC(CNC(C3CCC(C)C3)=O)C2)nc(Cl)nc2[nH]c(O)nc12 C(C(=O)N=c1ccn(C(F)F)[nH]1)C1N(C(C(CC)CC(C)C)=O)CC1 C1(CNC(C(C)=CC)=O)CCN(c2nc(C(=O)NC)cc(C)n2)CCC1(F)F CCCC(C(=O)N(C(C(=O)N(CC(O)(CC)CC)C)C1CC1)C)C(C)C C1(NC(CSC(C)C)=O)COC2(CCN(C(c3cc(Br)no3)=O)C2)C1 N(C1COc2c(Cl)cc(Cl)cc21)c1n(CCN(C)C)ncc1 N1(C(C2CCN(C(N(C)C)=O)CC2)=O)CCCC2(NC(C3CC3(F)F)=O)CC2C1 c1(C(=O)NC2C=CC(CNC(CCSCC(C)C)=O)C2)ccc(C#N)o1 Cc1oc(S(N)(=O)=O)cc1C(=O)NC(C)(CO)C(C)C c1(C(=O)NCC23N(C(C=CCOC)=O)CCC2CC3)ccc([N+](=O)[O-])cc1F N1(CC(=O)NCC(C)C)CCN(N2CCC(N3CCC3)CC2)C2CCCC12 C1(NC(C(=Cc2ccccn2)C)=O)CC2CCC(C1C)N2C(c1cncs1)=O CC(C(CO)NC(C1(C)CC1(F)F)=O)NC(c1cccn1C1CC1)=O c1(C(N(CCNC(=O)C(C#N)C2CC2)CC)=O)cnc2sc(C)c(C)n12 c1(NC(CC2CCN(C(C(C)(C)F)=O)C2)=O)cnc(Cl)cc1I CC1=C(C(=O)NCCC2CSCCN2C(c2cc3scc(C)c3[nH]2)=O)SCCO1 Fc1cc(CN2CCCCC2CCC2CCCN2)ncc1Br c1(OC)cc(Br)c(NC(=O)CC2CCCN2Cc2cnn(C(C)C)c2)c(Br)c1 C1(COC)CCCN1C(=O)CC1(CC(=O)O)CCC1 Cc1ccc(CCC(N2CCC(C(C)(C)NC(=O)CCSC3CCCC3)C2)=O)s1 N1(C(c2ccc(C(N)=O)s2)=O)CC2CCCC1C2CNC(=O)C(F)OC(F)(F)F Cc1cc(CO)oc1C(=O)NCCC(O)CNC(=O)Cc1cccnc1 C1(NC(c2nccc(CC)c2)=O)CC2C1CCN2C(c1cc(C(N)=O)co1)=O CC1CC(C)CN(C(C2COCCN(C(c3ccco3)=O)C2)=O)C1 C(C(C)(C)C#CC(=O)N(C)OC1CCCC1)NC(CC(C)O)=O c1(C(N(CC(CN(CCOCC(C)C)C)O)C)=O)cnn2c1CCC2 C=CCC(CC(F)F)C(=O)N1CC(NC(C2CCO2)=O)C1 N1(C(c2nc(C)c(C)[nH]2)=O)CC2(C1)CN(C(=O)C(C1CCCN(C)C1)(C)C)C2 c1(OCC(N2CCC(C(C)NC(=O)C(C)CN(C)C)CC2)=O)cc(Cl)ccc1Cl O=[N+]([O-])c1ccc(Cl)c(SCCCC2CCC2)c1 C1(CNC(C2(C#N)CCCC2)=O)CN(C(c2cncnc2C2CC2)=O)CC12CC2 CN1CCC(C(=O)NC2(CCNC(=O)C=CC3CCCCC3)CCCC2)CC1=O CCC(C(=O)NC1(CNC(=O)CNc2ccccn2)CC(OC)C1)C(C)C C(=O)(CCCS(N)(=O)=O)NC1CCN(C(c2cc(CC(C)C)on2)=O)C1 C1(CC(=O)NCC2N(C(C(CC)N(C)C)=O)CC(O)C2)CCC(C)(C)CC1 Cc1oc(Cl)nc1C(N1CC(O)(C(F)C(=O)N(C)CC2CCOCC2)C1)=O n1(CCC2(C)CC2)nnnc1C(c1cnc(C2CC2)s1)NCc1nccs1 N1(C(CNC(=O)NC)=O)CCCC2CN(C(c3nc(CF)cs3)=O)CCC12 CS(=O)(=O)CCC(=O)N1CCOC(CNC(c2ccc(-c3cccs3)o2)=O)C1 C1(C(=O)Nc2cccc(N(C)C)c2)C(C2CC2)CCN1C(c1cnn[nH]1)=O c1(CC(C)C(=O)N(C2CCCN(C(=O)CN3CCCC3)C2)C)ccc(O)cc1 C(=O)(C(C#N)=CC1CC1)NCC(C)NC(C1CC1c1ccco1)=O N1(C(C2C(=C)C2)=O)CC(C)C1C(=O)NCCCCNC(N)=O c1(C(=O)NC2CN(C(C3C(C)C3C)=O)C2)ccnc2[nH]c(O)nc12 c1(C(=O)NC2CN(C(C(c3c(C)cncc3)C)=O)C2)cnn2c1C(C)CCC2 C1(C(=O)NC2CCCCC2O)CCCN(C(=O)CC23CCCC2C3)CC1 c1(C(=O)NC2(CN(C)C(C3CCCN3C(c3cccs3)=O)=O)CC2)conc1C N1(C(CNC(N)=O)=O)CCCCCC(NC(=O)C(O)C(F)(F)c2ccccc2)C1 Cc1ccc2ncc(C(=O)NC3CN(Cc4cn(C(C)C)nn4)CC3F)n2c1 c1(C(C)NC(C2CCCSC2)=O)ccc(CNC(=O)COCc2nc[nH]n2)cc1 C1(C(=O)NC2C3(NC(c4[nH]cc(CC)c4)=O)CCC(C2)C3)CCC2(CCC2)CC1 c1(OCC(=O)NC(CNC(C2C(C=C)CC2)=O)(C)CO)cccc(F)c1 c1(CN2CCCC(C)(C(=O)NC(CC(C)C)CO)C2)c[nH]c2ncccc12 C#CC1(NC(C2(C)CCN(C(c3cn(C)nn3)=O)CC2)=O)CC2CCCC12 C(=O)(CC1COc2ccccc21)NCCOC1CN(C(C(C)(O)C2CC2)=O)C1 C#CCC(CC(F)F)NC(=O)COCCNC(C1CN(C)C(=O)N1)=O CCC(C)CC(=O)NCC1CC(NC(C2(n3cnnn3)CC2)=O)C(O)C1 c1(C(=O)NC(C(N2CCC(COC)C2)=O)C2CC2)ncn2ccccc12 c1(OCC)nccc(C)c1C(=O)NC1CC(C)CN(C(=O)Cc2cnccn2)C1 N1(C(CCc2cc(C)on2)=O)C2CCC1C(CNC(C1CC(F)(CO)C1)=O)C2 O=C(C1=CCCC1)NC(Cc1ccccc1)CCNC(C1(O)CCSCC1)=O CC1CC(C(N2CCCC(C)(CNC(=O)C=Cc3cccnc3)C2)=O)CC(C)C1 N1(C(CCc2ccc(OC)cc2C)=O)CC2CC(NC(=O)C(OC)OC)CC1C2 c1(CC(N2CC(OCCNC(C(CCO)N(C)C)=O)C2)=O)noc2ccccc12 c1(COC)nnc(CNC(c2nnnn2CCCF)c2cnco2)s1 C1(c2n(CCOC)nnn2)(Nc2cc(C)cc(F)c2)CCN(C(=O)C(C)C)CC1 c1(C(=O)NCC(C(C)C)NC(C(CCSC)N(C)C)=O)cc(Cl)ccc1Cl CC1CC(C(=O)NCC2(C)CC(NC(C3(C(N)=O)CCC3)=O)C2)=NO1 N1(c2ncnc(C)c2F)CCCC1C1CCCCN1C(=O)CC1CCCC1(F)F C1(CNC(C=CC=CC)=O)CC(O)CN1C(c1cn(C2COCC2F)nn1)=O c1(OC)cccc(C(CNC(=O)COC2CC2)NC(=O)CC2OCCC2(C)C)c1 n1(CC(=O)NCC(CC)NC(=O)CO)cccnc1=O CCC(C)(COC)C(=O)NC1CCC1NC(=O)Cc1cncnc1 C(=O)(CCC(F)(F)Cn1cc(CSc2c(O)ccc(F)c2Br)nn1)OC N(C(=NCC(=O)N1CCCC1)NCC1CCOCC1)C(c1cccc2ccsc12)C C=CCC(CC(C)C)C(=O)N1CCC2(CCN(C(c3cccc(Cl)c3N)=O)C2)C1 C1(c2nnnn2C)(NCc2c(C)con2)CCCCC1C CCCC(C#N)C(=O)N1CC(COC)(NC(c2csc3nccn23)=O)C1 C1(NC(=O)CC2(CO)CC2)C=CCN(C(C2(CO)CCOC2)=O)C1 C(C(CC(=O)NCCc1cccc(F)n1)C(F)F)NC(=O)OC(C)(C)C c1(C(=O)NCC(CNC(c2c(OC)nsc2)=O)O)c(C)cccc1C CCC(CC)CC(=O)NC12CCN(C(C3(SC)CC3)=O)CC1C2 C1(CC(=O)OC)CCN(N(Cc2nccn2C)CCCNC(N)=O)C2(CC2)C1 C(CCC(CC)CC)NC(C(CCNC(CC1(CC)CCC1)=O)N(C)C(C)=O)=O C1(CC(C)(C)C)CN(C(=O)CCn2cc(Cl)cn2)CCN1C(=O)CCC1(C)CC1 C(=O)(C(=O)C(C)(C)C)NC1C(NC(c2c(OC)cccn2)=O)CC1 c1(OC)ccc(C(=O)NCC2CCCC(CC)C2)nc1C C12(NC(=O)CCCCC3CC3)CCCC1N(C(=O)COc1ccsn1)CC2 c1(C(=O)NC(C(=O)NC(CCC)CCC)CO)ccc([N+](=O)[O-])o1 N1(C(C2(NC(C(CC)COC)=O)CCCC2)=O)CCSC2(CCC2)C1 C1(C(=O)Nc2ncc(C(C)=O)s2)CN(C(C2(O)CCOCC2)=O)CCS1 c1(OC(C)C)cc(F)cc(NNC(=O)OCCC2=CC3(CCC3)C2)c1 C1(NC(c2c(C)occ2)=O)CCCCC12CCN(c1cc(CC3CC3)ncn1)C2 C1(C(C)NC(c2cnc(CC(C)(C)C)s2)=O)CN(C(C2CC=CC2)=O)CCO1 N1(C(C2(CNC(c3ccn(CCC)n3)=O)CCCO2)=O)CCC(C)C1C c1(OC)cc2c(cc1C(=O)NC1CC(NC(=O)C(C)C)C13CCC3)OCO2 Cc1c(N)cc(C(N2CC(NC(=O)C(C)O)CC(C)(C)C2)=O)cc1N C1(C(N2CC3C(CNC(=O)CCc4cccc(-c5ccccc5)n4)(C3)C2)=O)CC12CCCOC2 C1(C(C)C)C(C(=O)N(C2CCCC(O)C2)C)CCN1C(C1CCN(C)C1)=O N1(C(C(CCC)C)=O)CCN(Cc2cnc3ccccn23)CC1C#N CC(C)CC(F)(F)C(=O)N1CCC(C2CC2)(CNC(=O)C(O)CN(C)C)C1 CC1CN(C)CCC1C(C(C1(N(C(=O)C(C)(C)C2CC2)C)CC1)=O)=O.C(CO)N N1(CC)CCOC(C(=O)NC2CN(C(c3ccc(C#N)[nH]3)=O)CC2O)C1 C1(CC#C)(C(=O)NCC(CC(=O)NC)OC)CCN(C(=O)CCOC(C)C)C1 c1(C(=O)NCCC2CC(NC(C3(O)COC3)=O)C2)nc(C2CC2(F)F)no1 C1(NC(C2OCCN(C(CCCCC=CC)=O)CC2)=O)CC2CCCC(C1)C2 C(=O)(CC(CN(C)C)C(F)F)N1CCC(CNC(c2cc(COC)sc2)=O)C1 c1(C(N2CC(NC(CCNC(=O)NC)=O)C(O)C2)=O)cccc(OC)c1C CC(C)(C(=O)NCCOCCNC(=O)CC1CC=CCC1)C1CCCC1 c1(CC)ccc(NC(C2(C)CCN(C(c3ncnn3C)=O)CC2)=O)cc1Cl Cc1c[nH]cc(C(=O)NC(C2(O)CCN(c3nccc(C(F)(F)F)n3)C2)C)c1=O c1(NC(C2CC(N(C(C=C)=O)C)C2)=O)ccnc2c1CCC2 N1(C(C2CC(=C)C2)=O)CC2CCCC(NC(=O)C3=C(Cl)CC3)C2C1 c1(C(N(CCNC(c2ccn(CC)c2C)=O)CC)=O)ccc2c(c1)CC(C)O2 N1(C(C(CC)C(C)O)=O)CCOC2(C1)CN(C(C1CCC(C3CCCO3)O1)=O)C2 CN1C(=O)Cc2ccc(C(=O)NC3CC(C)(NC(c4ccsc4)=O)C3)cc21 c1(C(C)C)cncc(C(N2CCCC(CCNC(C3(CO)CCCO3)=O)C2)=O)c1 N1(C(c2c(CC)non2)=O)CC(C)(CNC(=O)CC2CCCO2)CC1(C)C c1(C(=O)NCC(CC)(CC)NC(CCOCCOC)=O)ccn2nnnc2c1 c1(-c2nc(C)on2)cccc(C(=O)NCCNC(=O)CC2CSCCS2)c1 C12(C(N3CCCC3)=O)CC(CO1)N(C(=O)C(F)=CCN)C2.CO C(=O)(C(C)(CNC(C1(NC(N)=O)CC1)=O)CC)N(C1CC(CC)C1)C c1(NCc2c(OC)cccc2F)ncc(S(=O)(=O)N2CCC(C)(OC)C2)cc1Cl C1(C(N(C2CC3(CCC3)C2)C)=O)CC(C)(C)CCN1C(c1ccccn1)=O N1(C(C2(CC=C)CCCC2)=O)CCCC(N(CCO)C(c2ncn(C)n2)=O)C1 C1(C(=O)NC(COC)C2CC2)CN(C)CCN1C(C1C2CC3C(C2)C13)=O N1(Cc2ncc(CC)o2)CCCCC(NC(=O)CCOc2c(C)cccc2C)C1 C=CC(CCC)CC(=O)NCC1CCCN(C(C2C3CCC2CC3)=O)C1 CC1=NOC(C(N2CC(NC(C3(n4cc(Br)cn4)CCC3)=O)C2)=O)C1 C1(O)(CCNC(=O)C=CC2CCC2)CCN(C(=O)CC(=O)NCC(F)(F)F)CC1 CN1CC(=O)Nc2ccc(C(=O)NCc3cc(Cl)cc(Cl)c3)nc21 N1(C(C(=O)NC(C)C)=O)CC2CC(NC(C3COCCC3(F)F)=O)CC(C2)C1 C(=O)(C(C)C(F)(F)F)NCc1cn(C2CCN(C(C=C(C)C(F)F)=O)C2)nn1 n1(COC)ccc(C(=O)NC2(CCC(=O)N(C(C)CCSC)C)CCCC2)n1 CC1CC(=O)NCC1C(=O)NC1CCC(N(C)C(c2cscc2Cl)=O)CC1 C(N=c1[nH]c(Cl)ncc1Cl)C1C(C)CN(C(=O)C(F)Cc2ccccc2)CC1 N1(C(C(C)CN(C)C)=O)CC2CC(N=c3[nH]c(Cl)nc4[nH]cnc34)C2C1 N1(C(C2(C)COC(=O)OC2)=O)CC2CCC1CN2C(=O)C(F)C1CCOC1 c1(OCC)cccc(Cl)c1NC(C1(CNC(c2cc(Br)cc(Cl)c2)=O)CC1)=O C(C1=NOC2CCCC12)NC(C(C1CN(C(C2(Cl)CCCCC2)=O)C1)OC)=O n1(CC)nc(C)cc1CC(N1CCCCC1Cn1cc(-c2ccncc2)nn1)=O c1(CC(N2C(C(C)(C)CNC(=O)C(N)=O)CCC2)=O)cc(F)ccc1Br N1(C(CNC(c2ccoc2)=O)=O)CCN(C(C2COCCOC2)=O)C2CC12 C(N=c1[nH]c(N2CCC(C(F)F)CC2)nc(=N)[nH]1)c1nnc(C)o1 C1(C(=O)NC(C)CCNC(=O)CCN(C2CCCCC2)C)CC(C)(C)OC1(C)C O(NC(=O)CC(C)C1CCCN1C(C1(C)CC=CCC1)=O)CCOC(C)C CC1(C)CC(CC(N2CCC(C)(CCNC(=O)C=Cc3ccco3)C2)=O)CCO1 N1(C(c2c(C)c[nH]c2)=O)CC(C(C)(C)C)CC(CNC(=O)C(C)c2cccs2)C1 N1(C(CCC)=O)CCC(C2CN(C(c3ccc(N4CCCS4(=O)=O)cc3)=O)C2)C1 c1(CC)nc(C#N)cc(=NCC2CC(NC(C3CCCC4CC34)=O)C2)[nH]1 C1(CNC(C(C)=C(C)C)=O)CC2(CCC2)CN1C(c1ccccc1C1CCC1)=O N(C1COc2cccc(Cl)c21)C(c1cc[nH]c1C1CCC1)=O Cc1nc(O)c(Br)cc1C(=O)NCC1CCN(C(=O)C(C)C)C1(C)C Cc1nc(CC(=O)NCC2CN(C(c3cnc[nH]3)=O)CCO2)c(Cl)s1 c1(C(N2CCC2Cn2cc(C3(OC)CCOC3)nn2)=O)cc(-c2ccoc2)[nH]n1 N1(C(c2cc(C(=O)O)cc(F)c2)=O)CCCS(=O)c2ccccc21 CCCCC(C(=O)NC1CC(F)(CNC(=O)CC2CCN(C)CC2)C1)N(C)C C1(C(=O)NC(C)CN(C)C(C2CCN(C)C2=O)=O)SC2C=CC1CC2 N1(CCOCC)CCN(C2CCN(C(C3CCOCC3)C(N)=O)CC2)CC1 c1(C(=O)NC23CC2CN(C(c2ccncc2F)=O)C3)ccc2cccnc2n1 C(=O)(CC1=CCCCC1)N1CCC(C)(C(=O)NCC(F)(F)CC2CC2)C1 N1(C(CC(C)(C)SC)=O)CCOCC(CNC2CCN(C3CCN(C)CC3)C2)C1 c1(C(N(CC(O)CNC(=O)COCc2nccn2C)C)=O)cccc(OCF)c1 N1(C(C2CC(=C)C2)=O)CCCC(C2CCN(C(C3CCCC(F)(F)C3)=O)CC2)C1 c1(NC(COCC(CN(C2CCCN(C(N)=O)C2)C)O)=O)ccccc1[N+](=O)[O-] C1(C(=O)NCC2C=CCCC2)(CN(C)C)CN(C(=O)C=CC(=O)NC2CC2)C1 CC1CC=CCC1C(=O)NC1CC(CNC(c2ccc(CCN(C)C)cc2)=O)C1 Cc1nnccc1C(=O)NCC1(F)CC(NC(C2(C3CCCO3)CCCC2)=O)C1 N1(C(C2C(C#C)C2(C)C)=O)CCN(C(=O)CC2(NC(C)=O)CC2)CC1C C1(C2C(=O)O2)CCOC(C)(C)C1.C(CO)(CCO)NC(=O)OC(C)(C)C C1(C)(CNC(C(C)=C(C)C)=O)CCCN1C(c1sc(F)cc1Cl)=O C1(C(C)NC(c2cnc(C)s2)=O)CCN(C(c2ccnn2CC(F)(F)F)=O)CC1 c1(C(N(C2CCN(C(C(C)c3cccs3)=O)C2)C)=O)c(F)ccc(F)c1Cl Cc1ccc(C(=O)NCC2CCN(C(=O)C(O)C(F)F)C2(C)C)c(C2CC2)n1 CN1CCC(C(=O)NC2C3CCN(C(=O)Cc4sc(O)nc4O)CC23)CC1=O c1(C(=O)NC2CC(N(C(C(C)CC(C)(C)C)=O)C)C2)cnc2c(c1)NCC(=O)N2 Cc1oc(C#N)cc1C(N1CC2(CCC2NC(=O)C(C(C)C)n2ccnc2)C1)=O Cc1cccn2nc(C(N3CCOC(CN=c4cc[nH]c(C#N)n4)C3)=O)cc12 CC1(C)CC(NC(=O)CCOCC(F)(F)F)CN1C(c1ccc(F)c(CO)c1)=O C1(OC)CCC2(C(=O)N(CC(C)CNC(=O)C(C)Cn3ccnc3)C)CC12 c1(CCC(=O)NCC2(O)CCCN(C(C(C)=C(C)C)=O)C2)c(C)nc(O)nc1C C1(c2n(C)nnn2)(Nc2ccc(N3CC=CC3)cc2)CCCN2CCSCC12 C(=O)(N=c1cc[nH]c(C)c1C)C1N(Cc2c(C)cc(Br)cc2)CC(F)C1 c1(C(=O)NC2CCC(N(C)C(C3CCCC3(F)F)=O)CC2)c(C#N)cnn1C C1(C(=O)NCC2CCN2C(=O)COCc2ccncc2)(CC)CC1(F)F C(=O)(N(CCC(=O)N1CCCC1c1ccon1)OC)C1C(=C)C1 Cc1ccc2occ(CC(=O)NC3(CNC(C4OCCCO4)=O)CCOC3)c2c1 N1(C(CP(C)(C)=O)=O)CCCCCC1C(=O)NCCN1CCCCC1 C1(N(C=O)Cc2nc(CCC)sc2)CS(=O)(=O)C12CCOCC2 CCC(C)C(CC(=O)NCCSCC(C)C)NC(c1cnc(O)cc1C)=O N1(C(Cc2nc(=N)[nH][nH]2)=O)CCC(C2CC2)(NC(C2CCCC(=O)N2)=O)C1 c1(C(=O)NCC(CC(F)(F)F)NC(c2c(CC)nc[nH]2)=O)cc(C#N)ccc1C N1(Cc2onc(CC(C)C)n2)CC=C(CCNC(c2ccn(C(C)C)n2)=O)CC1 c1(OC)ccc(N=c2nc[nH]n3cc(Br)cc23)c(F)c1 Cc1n[nH]c(C)c1CC(=O)NCC1CC1NC(c1cn(C2CCOCC2)cn1)=O N1(C(c2c[nH]c(=NC)o2)=O)CC2CN(C(=O)CC3(CO)CCC3)CC2C1 C(C(CNC(=O)C(O)CN1CCCC1)S(C)(=O)=O)NC(c1c(OC)cncn1)=O C1(NC(c2cc(CC)no2)=O)CCN(C(c2[nH]nnc2CC)=O)CC1CC Cc1nn(C)c(C)c1C(N1CC2(CC2C(=O)Nc2cccnc2O)C1)=O CC1CCC(C(=O)N(C2CCCCC2N(C(=O)C=CC(F)(F)F)C)C)CC1 CC1(C)CC(C(=O)NCCCCNC(c2cnc(C3CCC3)s2)=O)CCO1 C(=O)(C1CCCn2nccc21)NC1CN(C(c2nc(C)sc2C)=O)CC(O)CC1 c1(CC)ncnc(CC)c1C(=O)N(C)CCN(C)C(c1cc(C(C)=O)cn1C)=O S(=O)(=O)(c1ccc(NCC2CCCCS2(=O)=O)cc1Br)N(C(C)C(C)(C)C)C C=CCC(C)(C)CCNC(c1c(CNC(=O)CC(C)SC)cnn1C)=O C1(OC)CC(NC(C23CC(C)C2C3)=O)CN(C(=O)C(C)(C)Nc2ccccn2)C1 CC1(C)NC(=O)CCC1N(C(=O)CCCCC(N)=O)C1CCCCC1 C(CCC(=O)N(C(C)C(=O)N(C)C(C)C1CC1)CCC)OCCC c1(OC)cc(C(N2Cc3nnsc3C2)=O)cc([N+](=O)[O-])c1Cl CC1CN(C(c2cc(Cl)ccc2F)=O)CCN(C(C2(c3ccn(C)n3)CC2)=O)C1 C(=O)(C(C)(F)C(=O)Nc1cccc(NC(C2CCSC2)=O)c1)OC C1(C(CCC)=O)CCCC(NC(=O)CCN2CC(Oc3ccccc3)C2)C1 C1(C(=O)NC2(CC(N3CC4C(COC)C4C3)=O)CC2)COc2ccccc2C1 c1(CNc2nccc(N=[N+]=[N-])c2)cccc2c1CCN(CCc1ccccc1)C2 N1(C(C2(COC)CCCO2)=O)CCN(C(c2ccn(O)c(=O)c2)=O)CC(C)(F)C1 CN1CC2C(C(N3CC(Cn4cc(CNS(=O)(=O)C5CC5)nn4)C3)=O)C2C1 N1(C(C2(C(N)=O)CC2)=O)CC(C2(NC(C3CCC(CCO)CC3)=O)CC2)C1 CCCC(C)CC(=O)NC1CCCC1NC(c1ccccc1CO)=O c1(CC(C)NC(=O)CCC(N)=O)ccc(CNC(C2CCC2(F)F)=O)cc1 c1(NC(C)=O)cccc(NNC(=O)c2cc(C)sc2-n2cccc2)c1 C1(O)(CNC(c2nn[nH]c2Cl)=O)CCN(C(c2ncncc2Cl)=O)C1 N1(C(CC(C)F)=O)CCCCC(CNC(c2sccc2C#N)=O)C1 Cc1c(C=CC(N2CCCN(C(c3ncncc3F)=O)CC2)=O)cnn1C C1(C2CCC2)(C(=O)NCC(C(=O)OC)Cc2ccncc2)CCC1 C1(C(=O)NCC2(F)CN(C(C(C(=O)OCC)(C)F)=O)C2)CCCC12CCOCC2 C(=O)(CC(C)(C)C(=O)OC)NCc1c(CNC(C(C(CC)C)C)=O)cccn1 C1(NC(CCC(=O)N(C(C)C)C)=O)CCC(C)N(C(C2CC3COCC3C2)=O)C1 Cc1nccc(C(=O)NCC2(CNC(C3CCN(C)C3=O)=O)CC23CCC3)n1 C1(NC(Cc2c(C)occ2)=O)CN(C(=O)CCOCC(F)(F)F)C2(CCOC2)C1 CC1CC(N=c2ccc(Br)c(S(=O)(=O)NCC(CO)C(C)(C)C)[nH]2)C1 Cc1cc(C)c2cc(C(N3CCCC(NC(=O)C(C)(C)CF)C(F)C3)=O)sc2n1 C1(NC(C2CC3(CC(OC)C3)C2)=O)Cc2ccccc2N(C(=O)C(C)CSC)C1 C(=O)(C(O)CC(N)=O)NC(C)(C)CC(=O)NCC(C)(O)Cn1cc(Br)cn1 C1(C(=O)Nc2cccc(CNC(C3CC=CC3)=O)c2)CCc2cncn2C1 C12(CNC(C(COC)O)=O)CCC(CC1)N(C(C1(C)CCN(C(C)=O)C1)=O)C2 C1(CC(N2CCC(CC#C)C2)=O)CC(C)(C)CN1C(=O)CCOCC1CCC1 C1(NC(CCc2cn(C)nn2)=O)CCC12CCN(C(=O)CCCCCF)CC2 N1(C(c2cnc(C#N)s2)=O)CC2CCC1CN2C(c1cnc2sccc2c1)=O c1(C(=O)NC(CC)CN(C(=O)C(O)CSC)C)cc(C)sc1Br CCCC(CC)CC(=O)N1CC(NC(c2ccc(N)c(N)n2)=O)C(C)C1 N1(C(CN(C(CC2OCC(C)(C)C2)=O)CC2CC2)=O)CCC2CCC(O)C1C2 Cc1cc(C(=O)NNC(=O)C2CC(=O)N(C)C2)c(C)n1-c1ccccc1N(C)C CCC(C)CCCCC(=O)NC1CCN(C(c2cnn3c2N(C)CC3)=O)CC1O CC1CN(C(=O)Cc2csc(NC=O)n2)CCCN1C(C1CC2CC1C2)=O c1(N2CC3(OCC(NC(c4ccnc(C)n4)=O)C3)C2)nc(Cl)nc(C)c1[N+](=O)[O-] c1(C(=O)NC2CC(NC(CC(COC)COC)=O)CC2O)cnc2cc[nH]c2c1 CCC(C)CCC(=O)N1CCC(NC(c2cnn(C3CCCC3)c2)=O)C(O)C1 c1(CCC)onc(C)c1C(=O)NCc1nc(CNC(c2cnc[nH]2)=O)cs1 CCC(C)C(O)C(=O)NC1CC(OCC(=O)NC(C(C)C)C2CCCC2)C1 N1(C(C(CO)N(C)C)=O)C(C(=O)NCCn2cc(CO)nn2)C2CC(O)C1C2 CCC(C(=O)NCC1CCN1C(=O)Cc1csc(S)n1)n1ccnc1 N1(C(c2c(C)oc(C(F)(F)F)n2)=O)CCN(C(=O)CCOC(C)C)C2CC12 N1(C(c2c(C)n[nH]c2)=O)CCCCC2(CCN(C(c3cc(CO)oc3C)=O)C2)C1 CC1CC=C(C(=O)NCc2ccnc(C(=O)NCc3ccco3)c2)CC1 n1(CCCC(=O)NC2(CNC(C(C)=C(C)C)=O)CCOC2)c(O)nnc1O c1(NCC(C)Cc2cnc[nH]2)ccc(S(=O)(=O)NCC2(S(C)=O)CC2)cc1F N1(C(CCc2n(C)ncc2)=O)CC(NC(C2(C(N)=O)CC2)=O)C(C2CC2)C1 c1(CNC(c2ccc(C(=O)OCC)cc2)C)ccc(OC)c(OC)c1 N1(C(C(C=C)(C)O)=O)CC2COCC2(C(=O)NCC(C)CN(C)C)C1 N1(C(CCN(C(=O)C2=NOCC2)C(C)C)=O)CCC(C)(C2CC2)CC1 C1(CNC(C2CC(S(C)(=O)=O)C2)=O)(NC(C2CCCCC2)=O)CC2CCC1CC2 c1(C(N(C)CCNC(c2csc(-c3ccccc3)c2)=O)=O)cncc2[nH]ccc12 C1(NC(C(CSCC)NC(C)=O)=O)CN(Cc2noc(C)n2)CC1C#N N1(C(C(C2CC2)SC)=O)CC(NC(=O)C(c2cccn2C)=O)CC(C)C1 O=C(CCCCCCCO)N1CC2CC2(C(=O)Nc2ccc(O)cc2Br)C1 CCC(C)(O)C(=O)NCC(c1ccccc1F)NC(=O)CC1CCC1 Cc1cc(C)c(OCC(N2CC(NC(=O)CN3CC=CC3)C3CC3C2)=O)c(C)c1 C1(CC(=O)NCC2(OC)CN(C(C3(O)CCCCC3)=O)C2)CCC(C)CO1 C1(C(N(CC(C)NC(C2C(=C)C2)=O)CC)=O)(OC)CCCCC1 c1(C(N2CC3(CN(C(c4c(C(N)=O)nccn4)=O)C3)C2)=O)cc(F)cc(Br)c1F N1(C(c2ccn(C)n2)=O)CC2OCCN(C(C3CC3C(F)F)=O)C2C1 c1(C(=O)OC)ncccc1SCCC1CC1.c12cn(nn1)CCN(C1CC1)C2=O C1(CNC(C2(O)CCSCC2)=O)CCCCC1NC(C1CCCCC1)=O N1(C(C(C)OCCOC)=O)CCCC(C)(NC(C2CCC(C(C)(C)O)CC2)=O)C1 N1(c2n(CCCOC)c(C3C=CS(=O)(=O)C3)nn2)CCn2c(C(C)C)nnc2C1 N1(C(C(C=C)OC)=O)CCC(F)(C(=O)NC23CCN(CC2)CC3)CC1 CC(C)CC(O)C(=O)NCC1(CCNC(C2CCC(CN(C)C)O2)=O)CC1 C1(C(=O)NCCCOCCNC(=O)COc2cccnc2)CCSCC1 N1(C(C(CCC)NC(C)=O)=O)CCC2(CCC(Nc3ccc(C)c(Br)c3)CC2)C1 CCC(CNC(c1csc(C(C)(C)C)n1)=O)(CC)NC(=O)CC1CCC12CCC2 N1(C(Cc2cc(C)sc2)=O)CC(C(=O)NC2CCOC(C)C2)C(C)(C)C1 CC1CCc2cc(C(N3CCC(F)(CNC(C4CC(F)C4)=O)CC3)=O)ccc2N1 c1(NCC(=O)Nc2ccc3c(c2)OCCCO3)nc2c(C(F)(F)F)cccc2s1 n1(-c2n(C)nnc2)nc(-c2cncc(Br)c2)nc1-c1ccnc(O)c1 c1(OC)cn(CC(N2CCCC(CN(c3cnc(F)cn3)C)C2)=O)c(C)cc1=O CCS(=O)CC(=O)NCC1(NC(=O)C(c2ccc(C)cc2)=O)CC1 CN1CCC(C(=O)NCCN(C(=O)COC(F)F)CCO)(NC(=O)OC(C)(C)C)C1 c1(CCC)nc(C)c(NC(=O)C(=O)NC(C)(C)CC(=O)OC)s1 C(=O)(C(C)(C)C(C)(F)F)NC1CCCC(NC(Cc2c(C)ocn2)=O)C1 N1(C(C2C(C=C)C2)=O)CCC2C(CCCN2C(c2ncccc2OC)=O)C1 C=CC1(C(=O)NCC(c2ccc(F)cc2)NC(C2CC2(F)F)=O)CCOCC1 N1(C(CC2(O)CCN(C)CC2)=O)CC2CC1CCC2NC(c1ncc(F)cn1)=O C(=O)(C(F)(F)F)N1C(C(=O)NCCCN(CCCOC)C2CC2)CC1 C1(C(C)NC(=O)CC(C)c2ccncc2)CCN(C(C2CC(F)C2)=O)CC1 Cc1csc2ccc(C(=O)NCCOCCNC(=O)C(O)C3CCCC3)cc12 C1(OC)CC(CNC(c2cnc(C3CC3)o2)=O)N(C(=O)C=CC2CCCO2)C1 C1(C)(COC)CC(NC(=O)C2=CCCCO2)CN1C(=O)Cc1ccsc1Cl C12(C(N3C(CCCNC(=O)CC4CC5(CC5)C4)CCC3)=O)CCCC1C2(F)F CCCCC(O)CCC(=O)NCCC1CCCN1C(c1cccc(F)c1C#N)=O c1(N(C)C)cncc(C(=O)NCCC2(NC(=O)CCc3cnn(C)c3)CC2)c1 N1(C(CC2CCC(NC(c3ccn(CC)n3)=O)C2)=O)CCC(O)(C(N)=O)C1 S(=O)(=O)(c1cnn(C)c1)N1CC(F)CC(NCc2c(OC)cccc2Br)C1 CC(C)C(C(=O)N(C)CC1(NC(=O)CC2CCC(C)CC2)CC1)NS(C)(=O)=O Cc1cc(C(N2CCC(NC(=O)COCC3CCCOC3)C(O)C2)=O)nc(O)c1 C=C(C)C(CC(=O)NC(c1ccc(NCCC2CCS(=O)(=O)C2)cc1)C)OCC c1(C(=O)NCC2OCCN(C(Cc3nc(C)oc3)=O)C2)ccc(F)cc1C(F)F C1(C(N2CC(NC(C3(OC(C)=O)CC3)=O)C(C)C2)=O)CCC(C)=C(C)C1 c1(CC)cccc(CNC(c2cccc(F)c2)Cc2ccncc2)c1F C(=O)(CC1=CCOCC1)NC1CC(C)N(C(=O)C=Cc2ccc(Cl)cc2F)C1 c1(OC)ccc(C(=O)N(C)Cc2ccccc2CNC(C2CC2(C)C)=O)nn1 C(=O)(C(CO)C(C)C)NCc1c(OC)cccc1.C12CCC(CC1)NC(=O)N2 C(=O)(C(CC(C)(C)C)OC)NC(C(=O)NCCCC=C)Cn1cncn1 N1(C(C2=C(C)OCC2)=O)CCCC2(CCCN2C(C2CC2(C)C)=O)C1 N1(C(c2cccc(SCCCC)c2)=O)CCCC(C)(NC(c2cnc[nH]2)=O)C1 CN1C(=O)OCC1C(=O)NC1(C)CCN(C(=O)CC(C)C2CCCCC2)C1 C1(C(=O)NCCNC(c2ccc(OC)c(C)c2)=O)CC2C=CC1C21CC1 C(=O)(C1=CC(O)C(NC(=O)CCCC2CC2)C1)OC N1(C(C2(C)CC(=C)C2)=O)CCC(NC(c2csc(C)c2Br)=O)CC(O)C1 N1(C(c2cc(C)sc2C)=O)CCOC2CN(C(C3CCC(C(N)=O)C3)=O)CC12 C1(C)(CNC(C(CCC)C)=O)COCCN(C(C2(C(F)F)CCCC2)=O)C1 CC(c1ccccc1Cl)=CC(=O)N(CCC(C(C)C)NC(=O)CC(F)F)C C1(CNC(C(CCSC)O)=O)CC(F)(F)CN1C(c1ccc(F)cc1C)=O N1(C(C(C)OC2CCCCC2)=O)CCC(N=c2[nH]cnc3cnccc23)C1 O=C1CC2C(C(=O)NCCC(F)(F)Cn3cc(CCCF)nn3)C2C1 C(=O)(C(C)C(=O)NC1CC(CC)(CC)C1)N1CC(N(C(COCCCC)=O)C)C1 C(=O)(CC(C)C(C)C)NC1CCN(C(C(CC)NC(c2ccccc2)=O)=O)C1 c1(CNC(c2c(C)cc(F)s2)=O)n[nH]c2c1CN(C(C1CC1F)=O)CC2 c1(C(=O)NCC(C2N(C(COCCC)=O)CCCC2)(C)C)nc(O)nc(O)c1N N1(C(CC2CCN(C(CC=C)=O)C2)=O)CCN2CCC1C2 Cc1nc(O)ccc1C(=O)NCc1ocnc1C(N1CCC(n2ccnc2)C1)=O CN1CCCC(N=c2ccnc(N3CCC(c4ccncn4)CC3)[nH]2)C1 CCC(C)C(C)(O)CNC(C1(N(C(=O)C(C)(C)C#N)C)CC1)=O Cc1cc(C(=O)NCC(C2CC2)N(C)C(c2ccc3c(c2)CC3)=O)cc(F)c1 C12(CNC(CCOCC(C)C)=O)CCC(CC1)N2C(C1CC1F)=O C1(C2CN(C(c3ccnn3CC3CCC3)=O)C2)(NC(C2CCC(=O)O2)=O)CC1 N(C(=NCCC1CCC1)N1CCC(OC2CCN(C)C2)CC1)Cc1scc(C)n1 c1(C(N2C(CNC(c3cccc(C#C)c3)=O)CC2)=O)nn(CC)cc1[N+](=O)[O-] C(C(C)(C(C)C)NC(=O)CSC(F)F)NC(CCCC)=O C=C=CCCC(=O)N1CCC(C2CCCCN2C(C2CCCC2)=O)CC1 C(=O)(CCCC(=O)NC1C2CNCC12)N1CC(CC#N)C1 N1(C(CN2CCC(C)C2)=O)CC(CNC(=O)C=Cc2nccs2)C2(CC2)C1 N1(C(COCCCC#C)=O)C2CCC1CC(NC(c1ccnc(C(N)=O)c1)=O)C2 C(=O)(CC(C)(C)C(=O)N1CCC(CNC(=O)C=Cc2ccnn2C)(OC)C1)OC c1(N(C(C)=O)C)ccccc1C(=O)NCCC(O)CNC(C1CC(CF)C1)=O CC#CCCC(=O)NCC(CCOC)NC(C1CC(F)(F)CS1)=O Cc1nc2c([nH]1)CN(C(C1CCN(C(=O)C(O)CC(C)(C)C)CCO1)=O)CC2 C1(NC(c2ccc(N(C)C)cn2)=O)CC(NCc2ccc(F)cc2F)C12CCC2 c1(CC)cccc(C(=O)NC2CC2CNC(=O)C(C)SC)c1N C(=O)(C1=C(C)CCCC1)N(CCN(C(c1cncc(OCC)c1)=O)CC)CC c1(C(=O)NCC(CCCC)NC(C2CC(CN(C)C)C2)=O)cc(F)ccc1C C(=O)(CCCCC(C)CC)NCCOCCNC(CC(C=C)(C)C)=O N1(C(C(CC)O)=O)CCC2(CCCN(C(=O)C(C)c3ccco3)C2)CC1 CC1CN(C(c2cc(CNC(=O)C=Cc3ccncc3)on2)=O)CCC1O c1(C(=O)NCC(CNC(C(C)Sc2ccc(C)cc2)=O)O)ccc(C)cc1O C1(CNC(C2CCCC23CCC3)=O)CCN(C(C2CCC3(CC3)C2)=O)CC1O N1(C(C2N(C(C)C)CCC2)=O)CC2CC1CC2NC(=O)COCc1ccncc1 C1(NC(C=C(CC)C)=O)(CNC(c2cnc(O)o2)=O)CC(C(F)(F)F)(OC)C1 C(=O)(C(C)CC(=O)N1CCCC(C)(NC(C2(c3ccccc3)CCC2)=O)C1)OC c1(CNC(C(N2CC(C#C)N(C)CC2)=O)=O)ccc2c(c1)OCCO2 N1(C(c2cc(OCC(C)C)ncc2)=O)CC2CN(C(c3cnc(Br)s3)=O)CC12 C12(C(=O)NCC3C(NC(=O)COC4CCCC4)CC3)CCC(CC1)C2 C1(C)(C(=O)NCC2N(C(c3cn(C)c(O)n3)=O)CCC2)CCCC1(F)F CC1(CNC(c2ccnn2C2CC2)=O)CCCN(C(c2ccc(Cl)nc2Cl)=O)C1 C1(C(N(CC(C)NC(=O)CC2(C)CC(F)(F)C2)C)=O)CCCN(c2nccs2)C1 N1(C(C2CCC(C)(C)OC2)=O)CC2CC1CN(C(c1cc(C(F)F)[nH]n1)=O)C2 CN1CCc2c(sc(N(C(=O)CC(O)CC(C)(C)C)CCNC(=O)CN)c2C#N)C1 C1(NC(c2ccc(SC)o2)=O)C2CC1CN(C(c1ccc(CN(C)C)cc1)=O)C2 C(=O)(C(C)CC(C)(C)C)NCCOC1CCN(C(Cc2c(C)cc(C)s2)=O)C1 N1(C(c2sc(Cl)cc2Br)C(=O)NCCOC)CCOC(c2ccccc2OC)C1 C1(C(=O)NC2(CNC(CCC=CC)=O)CC2)CCCC(C)CC1 c1(C(N(CC(CC)NC(=O)Cc2ccc(F)cn2)C)=O)ncc(Cl)cc1F C(=O)(C(C)CC(C)(C)C)N1C(C(=O)NCC(C(C)C)C)CC1 CCCCCOCC(=O)NC1CCC1NC(=O)CN(C)C(=O)OC Cc1cc(C(N2CCC(F)CC2)C(=O)NCC2CCCO2)n2nccc2n1 C(=O)(C1Cc2ccc(F)cc21)N(C1CC(NC(c2nccnc2O)=O)C1)C c1(C(N2CCCC(NC(C(CO)N(C)C)=O)C2)=O)nn(C)c(C(F)(F)F)c1Cl Cc1ccsc1C=CC(N1CC2(NC(=O)Cn3cc(C(F)(F)F)nn3)CC1C2)=O C=CCCCCN=c1[nH]c(N2CCC(F)(F)C3(CCOCC3)C2)nc2ccc(OC)cc12 c1(C(=O)NC2Cc3c(C)nn(C)c3CC2)nc2cc3c(cc2s1)OC(F)(F)O3 C1(CC)C(NC(C2CCCCO2)=O)CCN1C(=O)CN(CC)CC c1(C(=O)NC(C)CNC(C2CC(=O)N(C3CN(C)C3)C2)=O)ccc(S(N)(=O)=O)o1 CCCCCCCC(=O)NCC1CN(C(C23CC(C)(CCO2)C3)=O)CCN1C C1(NC(=O)Cn2cncn2)COCC1C1CC1.c12ccc(cn1)CNC2=O Cc1cc(C(=O)NCC2CCCC(CNC(=O)CCN3CCCCC3)C2)[nH]c1C C12(NC(C(C3CCN(C(COC(CC)C)=O)C3)F)=O)CCC(CC1)C2 c1(OC)ccc2[nH]c(=NC3CC=CCC3C)[nH]c(=NC3CC3C)c2c1 N1(C(C2(CC)CCN(C(c3cc(O)n(C)n3)=O)C2)=O)CCCC2(CCC2)C1C N1(CC(C)(C)NC(CC2(OCC)CC2)=O)CCN(C(C2CC(C)OC2=O)=O)CC1 N1(C(C2CC(SC)C2)=O)CC2CCC(C1)N2C(C1CCC(O)C1)=O N1(C(CCCC(=O)c2ccc(C)cc2)=O)CCCC(C2CCC2)CC1 c1(C(C(=O)Nc2nnc(CCOC)s2)(F)F)nnc2n1CCCC2 C1(C(N2CC(CNC(c3n(C=C)ncc3)=O)C2)=O)CC2COCC(C1)C2 C1(COC)CC(C)N(C(=O)NCc2ccc(N3CCOC(C)C3)cc2)CC1C Cc1nc(C)c(-c2nc(-c3cc(C)oc3C)nn2C2CCCCC2C)[nH]1 C1(CNC(CNC(=O)NC)=O)CC12CCN(C(C1CNC(=O)N1C)=O)CC2 c1(C(N2C(CCN(C(C(C)SCCCC)=O)C)CCC2)=O)cccc(CC)c1 C1(CCNC(=O)CSC(F)F)CCCCN1C(=O)CN1C(=O)CNC1=O c1(C(=O)NC2CN(C(c3nc(C)[nH]n3)=O)CC2(C)C)nc2cncnc2nc1O C1(CNC(=O)C(O)C2CC2)CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CCC1C(F)(F)F C(=O)(CCCC#CC)N(CCC(N1CCC(O)(CN(C)CC)C1)=O)CC#C CCCCCCCC(=O)NC1CN(C(=O)COc2cnn(C)c2)CC1C C1(NC(c2ccc(C3CCC3)nc2)=O)CCCC12CN(C(c1csc(Cl)n1)=O)C2 c1(OC)ccc(Cl)c(C(N2CC3(CCC3NC(=O)C(CN(C)C)N(C)C)C2)=O)n1 N1(CCNC(=O)C2=CCC2)CCC(NC(=O)Cc2ccc(OC(F)F)cc2)CC1 N1(C(c2c(CC)c[nH]c2)=O)CCCC(O)(CNC(=O)C2=CCC(C)CC2)CC1 N1(C(C2(C#N)CCC2)=O)CC2CCCC(C1)N2C(C1CC1C(F)(F)F)=O C1(CC)CN(C(=O)NCc2nccc(C(C)C)n2)C(C)CO1 N1(C(C=CCOC)=O)CC2CC(NC(=O)C(C)Oc3ccc(F)cc3)CC2C1 c1(C(=O)NCC2(NC(CC(C)N(C)C)=O)CC2)cccc(-c2ncon2)c1 C1(CC)CCCCN1C(=O)C=CC=C.C(CC(C)SC)NC(=O)C=CC(C)(C)C c1(OC)cc(C(F)(F)F)[nH]c(=NC(C)CN(C(=O)CC2=NNC(=O)C2)C)n1 N1(C(C2CN(CC)C(=O)N2)=O)CC2(CCN(C(c3ccccn3)=O)CC2)C1 CCC(C)C(=O)C(=O)N1CCCC(c2cn(Cc3ccccc3Cl)nn2)C1 c1(CC(=O)NCC(C)(C)NC(c2cc(C(C)=O)on2)=O)nnc(S)n1C C=CCCCC(C(=O)N1CCC(CC(=O)NC)C1)NC(c1cnn(C)c(=O)c1)=O C1(CNc2c(C)c(NC3CC4(C3)CC(N)CCS4)ncn2)C(C)(C)CCCC1(C)C c1(OC)cc(CC(=O)N(C)C(c2cn(C(C)C)nn2)C)cc(F)c1F N1(C(CC2N(CCC)CCC2)=O)CCN(C(=O)CCCOC(C)=O)CC(C)(C)C1 C#CC1(C(=O)NCC(=O)NCCC)CN(C(=O)Cn2nc(C)oc2=O)C1 Cc1cn2c(C(=O)NCCN(C(=O)CCCCCN(C)C)C)c(C)nc2s1 C(C)(CO)(C(=O)N(C)CCC1CCN(C(=O)C=CC2CCCCC2)CC1)OC CC#CCCCC(=O)N1CC2CC1CN2C(=O)CCc1ccc(C(=O)NC)cc1 C(CCCCCCCCC)(c1n(CC=C)nnn1)N(CC)Cc1ccc(F)c(F)c1 C1(N(C(C2CCOC2)=O)CC)CCCN(C(=O)Cc2cccc(OC(F)F)c2)C1 C1(CCNC(c2cnc(C)[nH]2)=O)CCN(C(C2CCC(=O)N2)=O)CCC1(F)F c1(C(=O)NCC(=C)Cl)conc1C(C)NC(=O)CC1CC2CC2C1 CC(O)C(C)C(=O)NC1CCCC1C(=O)OCc1cn(-c2ncccc2F)nn1 C1(N(C(CC)C)C(=O)CC2CC2CNC(=O)CSC(C)C)CC(O)C1 C1(CCC)CCOCC1(c1nnnn1CCOC)NC1CC(OC)C1SC c1(C(=O)NC2(CCO)CN(C(CSCCOC)=O)C2)cccc2c(C)c(C)[nH]c12 CC(C(=O)N(C1CC1)CC1CCCN1C(c1cc(-c2ccco2)c[nH]1)=O)S(N)(=O)=O c1(CNC(CN(C)C(c2ccc(-c3cc[nH]n3)s2)=O)=O)cc(F)ccc1F CC1CN(C(=O)C(C)(C)c2cnn(C)c2)CC1CNC(C1(C)CCC(=O)N1)=O CN1N=C(CC(=O)N2CCCC2CNC(c2cc3c(cn2)CCCC3)=O)CC1=O C1(NC(c2ccn(C(C)C)n2)=O)COCCC1NC(C1CCN1S(C)(=O)=O)=O C1(C2(C(N3CC(n4cc(CCCS(C)(=O)=O)nn4)C3)=O)CC2)(SC)CC(F)(F)C1 N1(C(C(CC)C(=O)OC)=O)CCN(C(=O)C(C)(C)CSC)C2(CCC2)C1 c1(C(=O)NCC2CC(NC(c3c(C)cc(O)nc3)=O)C2)cnc2n1C(C)CCC2 c1(C(=O)NC2CCN(C(c3cc(COC)oc3C)=O)C2)cnn2c1OCC(F)C2 C1(C(=O)N(Cc2cc(C)no2)C(C)C)CN(CCCC=C(C)C)CCC1O c1(CC)nc(C(N2CC=CC(NC(c3ccsn3)=O)C2)=O)c(C2CCOCC2)s1 Cc1cncc(NNC(=O)C2C(C)C2C)c1 CC1OCCCC1C(=O)NC1CCC(CNC(C2C(F)(F)C23CC3)=O)CC1 N1(C(CCc2ccc(OC)nc2)=O)CCCN(c2ncc(F)c(SC)n2)CC1C c1(C(=O)NCC(C)(C2CC2)NC(C(CC(C)(C)C)O)=O)cc(F)c(F)c(C#N)c1 N1(C(CN2CCC(C)C2)=O)CCCC(N(CCO)C(c2cc[nH]c2C2CC2)=O)C1 CC(CCCCNC(=O)C(=O)Nc1cccnc1)NC(c1nc(=O)n(C)[nH]1)=O Cc1ncnc(C)c1CC(=O)NCC1CCC(NC(=O)CC(C)C2CC2)CC1 c1(C(=O)NCC(C)(CO)NC(c2c(Cl)cc(C)s2)=O)cnc2ccccc2c1C N1(CC)CCN(CC(=O)N(C)CC2(O)CCN(C(C3CC3(F)F)=O)C2)C(=O)C1=O C(C)(C(C(C)C)NC(C1CC(F)(CO)C1)=O)NC(c1nc(COC)oc1)=O c1(CC)ncoc1C(N1CC(OCCC(=O)NC2CCCCC2)C1)=O C(=O)(C1CCCc2scnc21)NC1C(NC(c2c(C(C)C)ocn2)=O)COCC1 c1(C(=O)NCCOCCNC(CC(C=C)CC)=O)c(C)c2ccc(F)cc2oc1=O C1(OCC=C)CCN(C(=O)CCCNC(C23CSCC2C3)=O)C1 C1(NC(=O)C=CCn2cncn2)CC1C1CCCN(C(c2cnc(O)nc2O)=O)C1 C1(C(=O)NCCN(C(=O)Cc2csc(S)n2)C2CC2)CC(c2ccccc2)=NO1 C(c1ccc(Br)o1)=CC(=O)NCC(CNC(=O)C1=CCOC1)CO C1(C(N(C(c2ccccc2)C)C)=O)CC12CCN(C(C1C(C)(C)C1(C)C)=O)CC2 CC(c1ccccc1)=CC(=O)N(CC(=O)O)Cc1nc(CC(=O)O)cs1 Cc1cc(C)c(C(=O)NC(CO)C(C)NC(c2ccc(=O)oc2)=O)c(S)n1 c1(C(=O)NCCC(C)(C)NC(=O)CSS(C)(=O)=O)cccc2c1CCOC2 c1(C2C(C(N(CC(C)NC(=O)CC3CC=CC3)CC)=O)CCC2)ccc(F)cc1 C(=O)(C1CCSc2ccccc21)NC(CCN(C(Cc1cc(OC)no1)=O)C)C Cc1c(Cl)ccc(C(=O)NCCC2CN(C(C3(O)CC(C)(C)C3)=O)CC2C)c1N N1(C(C(C)CN2CCCCC2)=O)CCCC(NC(c2ccc(F)cc2F)=O)CC1 c1(CCN=C(NCC(=C)C)NCC(=C)Cl)c[nH]c2c(Br)cccc12 C1(C(=O)NCC2CN(C(C=Cc3ccc(C(N)=O)o3)=O)C2)CC2COCCN2C1 N1(C(C=C(COC)C)=O)CCN(C)CC1CNC(=O)CC(C)(C)N(C)C CCCN(OC)C(=O)C(c1cccs1)NC(=O)Nc1ccc(Cl)o1 c1(C(N2CCC(O)(CCNC(c3c(CC)cno3)=O)C2)=O)ccc2nncn2c1 CC(C(=O)N1CCC(F)(CNC(C2CCC(F)C2)=O)CC1)C(C)(F)F c1(OC)cnc(F)cc1C(=O)NC1C2CC1CN(C(c1cccn(C)c1=O)=O)C2 CC1CN(C(c2ccco2)=O)CCC1CNC(c1cc(Br)cnc1N)=O CC1CCN(C(C2CCC(F)CC2)=O)CC1CNC(=O)CC1CC(C)(C)CO1 C1(CNC(C(C)C2(O)CCC2)=O)CCC(NC(=O)C=C2CCSCC2)CC1 C1(C(=O)NC2CCC(CCC(=O)NCC(O)CCOC)C2)(CC)CCOC1 C1(C(=O)NC(c2cnn(C)c2)CC)CCCC1CNC(C1CCNC1=O)=O C1(CNC(c2[nH]cc(CC)c2)=O)CN(C(=O)C(C)(C)CCOC)CC12CC2 N1(C(C2C(Cl)(C(=O)OC)C2)=O)C2CCC1(CNC(=O)CC1=CCCC1)CC2 c1(SC)nn(C)c2nc(C)c(CCC(=O)N(c3cncc(Cl)c3)C)c(C)c12 CCC(CC(=O)NC1(CCC(=O)OC)CCC1)C(C)(C)C c1(C(=O)NCC23N(C(c4ccc(N)c(Cl)n4)=O)CC(C2)C3)cnc2[nH]cnc2c1 N1(C(C(C2(O)CN(C(c3ncn(CC)c3)=O)C2)F)=O)CC2(CCCCC2)C1 c1(CC)cnc(Cl)[nH]c1=NC1CC(NC(C2CCC(C)(C)O2)=O)C1 C=CC(C)(O)CC(=O)N(CC)CC1CCN(C(=O)C(C)C(C)O)CC1 N1(C(c2cc(C)[nH]n2)=O)CC(NC(C2CCCC2C2CC2)=O)C(C)(C)C1 C(=O)(C(O)CCC(C)(C)N)C(Cc1c(CNC(CC(C)C)CO)cccc1)=O c1(CCOC)cnn2ccccc12.C12(c3nnnn3C3COC3)CN(C1)C2=O c1(OCCC(C)C)cccc(CNC(=O)C(C(C)C)C2CCC2)c1 N1(C(CC(C)SC)=O)CC(F)(F)CC1(C)CNC(=O)C(C)=C1CCC1 C1(C(N(C)CC2(CNC(=O)CCC3CCCCC3)CC2)=O)CCNC1=O N1(C(c2c(CC)sc(=N)[nH]2)=O)CC(O)C(O)C1CNC(c1coc(COC)n1)=O C(C(F)(C(=O)N1CC(C)OC(C)C1)C(C)C)NC(c1cc(C)cc(F)c1)=O c1(C(N(CCC(=O)N(C2CC2C)C)CC#C)=O)cnc(OC)nc1 CC1CCC(C)N(C(=O)CCCCN(C)C(C2C3CN(C)CC23)=O)C1 c1(C(N2CCC(CC(C)NC(CCCC=C)=O)CC2)=O)c(C)cccc1N C#CCC(CC(F)F)OC=O.C(=O)(C(C)=C1CC1)N(CC1CCC1)CC c1(SC(CS(C)(=O)=O)CO)nc2ccc(Cl)cc2o1 c1(C(=O)NC(CC2CN(C(CCC(=O)NC)=O)C2)C)c(F)cc(Cl)cc1F c1(C(C(N2CC(NC(=O)CC(F)F)C(O)C2)=O)O)ccc(Cl)c(Cl)c1 C(=O)(C1=C(Cl)CCCC1)N1CC2C(CNC(CCc3c(OC)cccc3)=O)(C2)C1 Cc1sc(C(=O)NC(CNC(=O)C(C)OC2CCCCC2)C(C)C)c(C)c1C c1(OC)ccc(Cl)c(NC(=O)CC(C)(C)N)n1 C1(C)(C(=O)OC)CN(C(=O)C(N)CCc2cn[nH]c2)C(C)(C)C1 C#Cc1ccc(C(=O)NC2CN(C(C3(O)CCC(C)CC3)=O)CC23CC3)cc1 N1(C(=O)NCCCCOC)CCC(NC2CCCC2c2ccccc2)CC1 Cn1cc(C(=O)NCC(C)(C)CO)c2cc(-c3ccnc(CO)c3)ccc12 c1(CC)cc(C(=O)NC(CNC(c2ccncc2C(F)(F)F)=O)CC)c(C)o1 CC1(C)COC(CC(N2CCC(O)C2NC(=O)OCc2ccccc2)=O)CO1 C1(O)(CC)CCCN(C(=O)C(CNC(=O)C(C)NC=O)OC)C1 c1(C(=O)NC2CC3(CN(C(C4CC(C)CC(C)C4)=O)C3)C2)cc(S(C)(=O)=O)co1 C(C)(N=c1[nH]c2cccc(Br)c2o1)C1CCCN(C(C2C(C(=O)OC)C2)=O)C1 C1(C)(CNC(CC(C)F)=O)CN(C(c2ccc(-c3cn[nH]c3)cn2)=O)C(C)(C)C1 c1(OC)ccc(CC(N2CCC(NC(=O)C(C(C)(C)C)SC)C(O)C2)=O)c(F)c1 c1(OC)cc(C(N2CC(N(C(=O)C(O)C(C)SC)C)C2)=O)c(Cl)cn1 C(=O)(N=c1[nH]oc2cc(Br)ccc12)C1CC(SCC)C1 C1(NC(C2CN(C(COCCCOC)=O)CC2(F)F)=O)CCN(C)CC1C#N CN=c1nc(N2CC(F)(F)C(F)(F)C2)[nH]c(=NCc2cc(=O)cc[nH]2)[nH]1 n1(CCC(=O)NCCCN(C(C2(CC(F)F)CC2)=O)CC)ccccc1=O C=CC1OCCC1C(N1CCCC1CC(=O)NC(C)C(=O)OCC)=O Cc1cn2c(n1)CCC(C(N1CCC(NC(C34CCCCC(F)(C3)C4)=O)C1)=O)C2 C1(NC(COCC(C)C)=O)CN(C(c2ccc(OC(C)C)cc2Cl)=O)CCC1F CCC(C(=O)OC)C(=O)N1CCCC(CO)(CNC(=O)CCc2ccncn2)C1 C1(C(N2C(C(=O)NC)CC2)=O)CN(C(C2CC(=C3CCC3)C2)=O)CC1C(C)C C1(Cc2cn(C(COCC)C(=O)NCC(C)(C)C(F)(F)F)nn2)CCc2ncnn2C1 N1(C(C(c2ccc(C)s2)C)=O)CCN(C(c2cccc(O)c2C)=O)C(C)C1 C1(C(=O)NC(CNC(c2c(C(C)C)nn(C)c2)=O)C)CC2(C1)CC1(CC1)C2 C1(C(N(C(CNC(=O)Cn2nnc(=N)[nH]2)C2CC2)C)=O)CNC(=O)N1 N1(C(c2ccccn2)C(=O)NC)CC2CCCCC2(C(=O)ON2CCOCC2)C1 Cn1c(C(=O)NCC2CC(CNC(=O)CNC(=O)NC3CC3)CO2)nnc1S c1(CCC(=O)NCC(C)(C2CC2)NC(C2(CC)CC2)=O)cccn1C C(=O)(C1=Cc2cc(OC)ccc2OC1)N1CC(C)(NC(CCOCCOC)=O)C1 C1(CNC(C(C)NC(N)=O)=O)CN(C(=O)C(C)OCCN(C)C)CC1C(F)(F)F N1(C(CSCC)=O)CCC(C(=O)Nc2cncc(OC)c2)C1(C)C c1(C(=O)NC2C(CNC(C(c3cncn3C)OC)=O)C2)ccc(CC#N)cc1 Cc1cnc2n1CCC(C(=O)Nc1cccc(-c3cn4ccsc4n3)c1)C2 c1(OC)ccc([N+](=O)[O-])c(N(C(C)CNC(=O)C(C(C)C)NC(N)=O)C)c1F C(=O)(C(C)C(C)n1cccn1)NC1(C)CN(C(C2(CCC)CC2)=O)C1 C(=O)(C1=NOC2(CCC2)C1)N1C2CCN(C(c3n(C)cc(C(N)=O)c3)=O)CC2C1 Cc1ccsc1C(=O)NCC(C(=O)N(C)CC1(F)CCCC1)N(C)C N1(C(CCN(CC)CC)=O)CC(OC)CC(NC(=O)C(CCC)OC)C1 c1(C(=O)NC(C2CN(C(=O)CC3CCCC3)CCO2)C)cc2ccc(Cl)cn2c1 N1(C(COCCCOC)=O)CCC2(C=C(C(=O)Nc3cnc4c(c3)CCC4)C2)C1 CCC(CCOC)C(=O)N(C)CCOCCCN(C(=O)Cc1sccc1Cl)C C1(NC(COCCCC)=O)CCN(C(C2CCCC2C2CC2)=O)CC1CO c1(OC)cc(OC)c(N)c(C(=O)N(C)CC2CCN(C(=O)CSC)C2)c1 N(C1c2ccccc2CC1NC(c1cscc1Br)=O)C(COCC#C)=O N1(C(C(=O)NCCCOC)C2CC=CC2)CCCC2(CC(O)C2)C1 C(=O)(CCCCC(C)(C)C)N(CC(C)C(N1CCS(=O)(=O)CC1)=O)C C=CC(C)C(C)C(=O)NCC1(NC(c2csc(Cl)c2Cl)=O)CCCC1 c1(NC(C2N(Cc3ccc(N(C)C)o3)CC2)=O)cnc(N2CCCCC2)nc1 Cc1nc(Br)oc1C(=O)NC1COCCC1NC(=O)C(C1CCOCC1)O c1(C(=O)NCC(C2CCC2)NC(C2CC23CC3)=O)cccnc1 c1(C2(C(=O)NC(C(C)NC(=O)CNC(C3CCC3)=O)C)CC2)cccc(Cl)n1 c1(CC(=O)N(CC(Cc2ccccc2)NC(C(C=CC)O)=O)C)sc(C)cc1C c1(OCC)nc(NC2CCN(C(=O)CN3CC4CCC3C4)CC2C)ncc1C N1(Cc2nc(CCC)sc2)CC2C(NC(c3cc(C4CC4)ccn3)=O)C2C1 c1(C(N2CCCC(CNC(=O)C(C3CCOCC3)F)C2)C)ccccc1F N1(C(c2c(C)n[nH]c2C)=O)CC2CCC(N(C(=O)CSc3ccncc3)C)C2C1 C1(C(=O)NCC(=O)NOC)(SC)CN(C(=O)C(C)OC(C)=O)C1 CCCC(C)(C)CC(=O)NC1(CNC(c2ccnc(Cl)c2O)=O)CC1 c1(C(=O)NC2CCCN(C(C(CC)n3ccnc3)=O)CC2)cccn2nncc12 CCC(CC)C(C)C(=O)NCC(C1CC1)N(C(=O)C=Cc1cc(F)cc(F)c1)C C1(NC(Cc2cccc(C)c2)=O)CCN(C(c2ccc(C)[nH]2)=O)CC1C N1(C(COCCC)=O)CC(NC(c2cnn(C)c2C)=O)C(n2cccn2)C1 c1(C(N(C2CN(C(C3C4COCC34)=O)C2)C)=O)cnc2c(c1)CNC2=O N1(C(COC(CC)C)=O)CC(O)(C2(CNC(=O)COC(F)(F)F)CC2)C1 N1(C(C(=O)Nc2scc(-c3ccc(C)c(C)c3)n2)=O)CCOCC12CCOCC2 CC1CN(C(c2ccc(CS(C)(=O)=O)o2)=O)CC1NC(C1(C(N)=O)CC1)=O c1(C(=O)NCC2(NC(c3ccnc(S)c3)=O)CC2)cccc2cnnc(O)c12 c1(C(=O)NC(CC(C)NC(c2cc(OC)n[nH]2)=O)C)cc(O)nc(N(C)C)n1 Cc1cccc(C)c1CC(=O)NCC1CCC1NC(=O)CCCN(C)C N#CC1CN(C(c2cnc(Cl)s2)=O)CCN1C(c1cc(Br)cc(Br)c1F)=O C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)N1CC(C2CN(C(C3C(OCC)C3)=O)C2)C1 CCC(CC)CCCNC(=O)NC1CC(CF)C1 c1(CC)csc(C(C)NC(C2(c3ncc[nH]3)CC2)=O)n1 CC(CC(=O)NC(C)C(CO)NC(C12CCC(CC1)CO2)=O)C(F)(F)F N(C1CCc2cc(CNS(C)(=O)=O)ccc21)CC1(CCN=[N+]=[N-])N=N1 C1(CNC(C2CC(c3ccccc3)O2)=O)CN(C(=O)CSC(F)F)CCCO1 CCCCC(C(=O)NC1(C)CCN(C(c2ccsc2-n2cnnn2)=O)C1)C(C)C CCC(CNC(=O)C(C)(C)C(C)NC(C1CCCN1C(N)=O)=O)(CC)CO CON1CCC(CC(=O)N(C2CN(C(=O)C(C)CC(N)=O)CC2O)C)CC1 C(C(C)(C)C(=O)NCC1(OC)CN(C(=O)CC(C)N(C)C)C1)OCC c1(C(N2CC(O)CC(NC(c3ccccc3F)=O)C2)=O)cc2cccc(F)c2o1 c1(-c2cn(C(COCC)C(=O)N3CCC(SC(C)(C)C)C3)nn2)cc(C)nn1C C1(N(C(=O)CC23CC(CCO2)C3)Cc2ccsc2)CC2(C1)CN(C(=O)CC1CC1)C2 Cc1ccc(F)c(CNC(C2CSCCN2Cc2ccc(Br)cc2I)=O)c1 CC1CC(C(=O)NC(CNC(C2(CCO)CC2)=O)C2CCC2)C1 c1(C(C)C)nnc(C=CC(=O)NCC2CCCC2NC(=O)C(C)(C)F)o1 C#CCCCCCC(=O)N1CC2(C1)CN(C(c1cc(C)n(CC)c1C)=O)C2 c1(OCC)ccc(F)c(C(N2CCC(NC(C3CN(CC)C3)=O)C(F)C2)=O)c1N CCC(C)C(=O)C(=O)N1CC2(CC2)CC1CC(N1CCC(O)C1CC)=O C(=O)(C1CCCc2cncn21)N1CC(N(C(c2c(CC)nns2)=O)C)C1 O=C1CC2(C1)CC(C(N1CCC(F)(C(N3CCCCC(CO)C3)=O)CC1)=O)C2 CN1CC2OCCN(C(C3(NC(=O)C(O)C(F)(F)F)CC(O)C3)=O)C2C1 N1(C(c2cn(C)nn2)=O)CC(C)(NC(CCOC2CN(C(C)=O)C2)=O)C1 CCC(C)C(C(=O)N(C1CN(C(c2cc(O)ncn2)=O)C1)C)NC(C)=O N1(C(=O)C2=CCOCC2)CCCC2(CCN(c3nc(Cl)nc4c3CCC4)C2)C1 c1(NC(C2CC2NCc2cnc3cc[nH]c3c2)=O)nc2c(O)cccc2o1 CC(C)(C)C(CC(=O)NC1(CO)CN(C(C2Cc3nncn3C2)=O)C1)C(F)F c1(N2CCC(O)C2)cccnc1N1CCCCC1.C1(NC=O)CN(CC2CC2F)C1 C#CCC(C)(C(=O)NC(CO)C(C)(C)CO)NC(=O)Cc1ccc(O)cn1 c1(C(N2CCC(C(CNC(C=CCOC)=O)C)CC2)=O)ccc(F)c(N)c1 N1(C(CCOCCCNC(C(=Cc2ccco2)C)=O)=O)CC(O)CC1C N1(C(c2n(CC)ncc2Cl)=O)CC2CN(C(c3cc(C(C)=O)cs3)=O)CC2C1 CC1CN(CC2CC=CCN2Cc2ccccc2)CCC1Nc1ncc(Cl)c(O)n1 CC(COc1ccccc1Cl)N=c1[nH]c2c(c(=NCCSCCO)[nH]1)CSC2 S(=O)(=O)(C1COCC1O)N1CCOCC(C(=O)NCC2CCCCO2)C1 Cc1c(-c2ccccc2F)o[nH]c1=NC(=O)C1C2COCC12 c1(C(N2C3CCC(CCNC(C(CC#C)O)=O)(C3)C2)=O)c(C)ccc(C)c1N CCCCC(O)CC(=O)N1CC(F)(F)CC1CNC(=O)Cc1cccnc1Br N1(C(C2(CNC(c3c(C)nccc3)=O)CC2)=O)CCN(C)C(C)C1 c1(CNC(c2nc(Cl)cs2)=O)coc2ccc(F)cc12 C=CC(CCC)CC(=O)N1CCN(C)C(C(=O)NCc2cc(OC)ncn2)C1 c1(N2CC(C)CC(C)C2)ncccc1S(=O)(=O)NCc1c[nH]c(=N)s1 CC(C)(C)C(C(=O)NC1CC(CCNC(C2CC3(CC3)CO2)=O)C1)NS(C)(=O)=O Cc1ccc([N+](=O)[O-])c(NCC(CC(C)C)NC(C2CCc3nnnn3C2)=O)c1 S(=O)(=O)(c1cccnc1OC(F)F)NC(c1ccncc1)C N1(CC2C(C)CCC2)C(=O)CCN(CC(c2ccccc2)(F)F)C1=O c1(C(N2CC(O)(CC(N3CC(O)(C(C(=O)OCC)F)C3)=O)C2)=O)cnc(C)n1C CCC(C)(C(=O)NCC(F)(F)Cn1cc(-c2ccc(F)cc2F)nn1)C(F)F c1(-c2cn(C3CC4(C(=O)NCCCC(=O)NC5CCC5)C3C4)nn2)cncc(Br)c1 C1(C(N2CC(C)OCC2)=O)CC(F)CN(CC2(C)CCS(=O)(=O)C2)C1 C1(NC(CCCCCC=C)=O)COC2(CCCN(C(=O)CC3CCCC3)C2)C1 c1(CN2CCC(N(C)C(c3cc(N(C)C)cc(Cl)c3)=O)C2)cnn2c1NCCC2 CC1CCc2nc(C(=O)NC3CC(CNC(c4ccc(F)c(Cl)c4)=O)C3)cn2C1 C(=O)(C1=Cc2ccccc2OC1)NC(Cc1cccc(OC)c1)C(=O)O C1(CNC(=O)CC2CSCCO2)CC2CC2N1C(=O)C=Cc1ncc[nH]1 C(=O)(CCCCCc1ccccc1)NC(CNC(C(C1CCCC1)OC)=O)C(C)(C)C C1(CNC(C(CC)N(C)C)=O)CN(C(=O)COC(C)(C)C(F)(F)F)CC12CC2 CC1(C)C2CCC1(C(=O)NCC1(NC(C3CC4CC(=O)C3O4)=O)CCC1)C2 C1(CN(C(=O)CCC2(C#N)CCC2)C)COCCN1C(C1CC(OCCF)C1)=O c1(C(=O)NCCN(C(C=C(COC)C)=O)C(C)C)cnc2c(F)ccc(F)c2c1 c1(CC)c[nH]nc1C(=O)NCC1CCCN1C(C12CC(OC)(C1)C2)=O Cc1cc2c(N3CCC(CC(N4CC([N+](=O)[O-])C4)=O)C3)nccn2n1 C12(NC(C3CCC(CC)O3)=O)CCC(CN(C(C3CN4CCC3CC4)=O)C1)C2 S(=O)(=O)(c1ccc(Cl)cc1)NCC(=O)NC1C(CNC(CC(C(C)C)C)=O)CCC1 CN1CCN(C(C2CNC(=O)N2)=O)CC1C(N1CCOCC1C1CCC1)=O C1(C(=O)NC2(C)CCN(C(=O)CC3CC4(CC4)CO3)C2)CC2(CCOCC2)C1 c1(-c2ccc(-c3ccc(NC(c4ccccc4)=O)cc3)nc2)ccnc2ccccc12 c1(NC2(CNC(C(C)=C(C)C)=O)CC2)ncnc2c1ncn2-c1ccccc1 c1(CNC(C2(C(C)=O)CCC2)=O)ncccc1C(N1CCC1CO)=O C1(NC(C=Cc2cn(C)nc2)=O)CCN(C(C2C3CCCC23)=O)CC(O)C1 c1(C(N2CC(NC(c3cc(CC)ncc3)=O)C3C2C3)=O)cc(N)cnc1Cl CC1CC2(CC(C(=O)N(C)CCNC(C3CCCS3(=O)=O)=O)C2)C1 n1(CC)ccc(CCNC(=O)C(C2CCC2)NC(=O)CN(C)C(C)C)n1 n1(CC)nc(C)c([N+](=O)[O-])c1N1CCN(C(c2cccc3c2OCO3)=O)CC1 c1(C(=O)NCC2C(NC(=O)Cn3nnc(=O)[nH]3)CCC2)c[nH]cc(Cl)c1=O N1(C(c2c(COC)ccs2)=O)CC(N(C(=O)CC2CCCC23CC3)C)C(O)C1 C1(SC(C(C)NCCSC)C)CCCN(c2cccs2)C1=O c1(CNC(CCN(C(=O)CCC2CCCO2)CC#C)=O)cn(CC=C)nn1 CONC(=O)C(Cc1cn[nH]c1)NC(=O)C(C)(F)c1ccon1 C1(CC(=O)N(CCCC(=O)OC)C)C2CCC(C2)N1C(C12CC(C)(CCO1)C2)=O N1(CC(C)(C)NC(CC2C(C)C2)=O)CCN(C(=O)CCc2ncccn2)CC1 N1(C(C(CC)(F)F)=O)CCOC2(CCN(CCOCC(F)(F)F)CC2)C1 N1(C(C=COCC)=O)CC(CNC(=O)CC2CCOCC2(C)C)CC12CCC2 CC(C)CC(C)CC(=O)N1CC(C2(Nc3nccc(C#N)n3)CC2)C1 c1(N(CCCCC(C)C)C)nc(=NCC2(CO)CCCO2)[nH]c2c1COC2 C(=O)(C1=CCOCC1)NC(CCOC)C(=O)NCc1nccs1 N1(C(COc2ccc(C)cc2)=O)CCCC(Nc2ncc(C3CC3)cn2)C1C C=CCCC(CC(C)C)C(=O)NC1CC2CC(NC(c3ccccc3)=O)C2C1 Cc1nnc2c(C(N3CCOC(CCNC(=O)COC(C)C)C3)=O)cccn12 c1(C(C)=O)ncc(C(=O)NCCCNC(=O)Cc2ccc(C)s2)s1 c1(CC(=O)NCC(C(C)(C)C)NC(CCCCN(C)C)=O)ncn2c1CCCC2 CC1(C)CC(CNC(=O)CCC(=O)c2cccnc2)CN1C(C1(CN)CC1)=O C1(CCC(=O)NCC(C)CN(C(=O)CSCc2ccccc2)C)CCC(O)CC1 N1(C(c2c(Cl)ccc(N)c2)=O)CCC(NC(c2ccc(CO)s2)=O)C2(CCC2)C1 c1(C(C(=O)OCC(F)(F)F)OC2CCSCC2)ccccc1 C(c1ccc(C(F)F)o1)=CC(=O)N(CC(C)NC(=O)COCC1CCCO1)C C1(C(=O)NCC23CC2CN(C(C2(O)CCSCC2)=O)C3)CC2C=CCC(C1)C2 CN1CC(C)(C)CC1C(=O)NCC1=CCN(C(c2ccc(=N)[nH]c2)=O)CC1 C1(C(=O)NCC2N(C(CN3CC(CC)C3)=O)CCCC2)CCc2n[nH]c(C)c2C1 C(C(C)(C)C#CC(=O)NCc1cnc(C(C)C)[nH]1)NC(C1C=C(C)CS1)=O C(C1C(C(=O)NCCCCC2CN(C(=O)Cc3nocc3C)C2)C1(C)C)=C(C)C C1(C(N(C2CCCCC2)CCNC(c2cccnc2O)=O)=O)CCCC(F)C1 c1(OC)cc(F)ccc1C(c1nnnn1C1CC1)NC1(c2ccccc2C)CC1 Cc1c(C(=O)NCC23CCC(CC2)C(C)(C)O3)n(C)c2ccccc12 C(=O)(C1=NNC(=O)C1)NCC1CCC(NC(C2CCC(C)CC2)=O)C1 c1(C(=O)NCCN(C(=O)C(C)CSC)CCOC)cc(C)ccc1C1CC1 Cc1nc2ccc(Br)cn2c1C(=O)NC(C1CCN(C(=O)C=C2CC2)C1)C C12(CO)CCCN(C1)N2.N1(C(=O)C=O)CCN(C(=O)C2CC2)CC1.c1(CO)ccccc1 c1(C(N2C(CNC(C3CNC(=O)N3)=O)CC(O)C2)=O)nccn2cnnc12 C(=O)(CCC1=CCCCC1)NC(C(=O)N(CC(=C)C)C)CC(=C)Cl N1(C(COCC=C)=O)CC(CNC(c2cnc(C)nc2C)=O)OC(C)(C)C1 C1(NC(C(c2cn(C)nc2)O)=O)CC(NC(C2CSC2)=O)CC1O CCC(CC(=O)N1CCOC(CNC(=O)CC2(c3ccon3)CCC2)C1)C(F)F N1(C(c2cccc(C#C)c2F)=O)CCCC2CN(C(=O)CN(C)C)CC12 C(N=c1cc[nH]cc1[N+](=O)[O-])C1CCN(C(c2cc(C)sc2C)=O)CC1C S(=O)(=O)(c1ccsc1C#N)NCC(C)(CO)OC Cc1c[nH]c2ncc(C(=O)N(C)CCN(C(=O)C3=NOC4(CCC4)C3)C)cc12 N1(C(C(=CC2CCCC2)C)=O)CCC(C)N(C(=O)CSCc2cscn2)CC1 C=CC1(CC(=O)N(C2(C)CC2)C)CN(C(=O)COC)C1 N1(CC(=O)NC2(CNC(c3ncc(C)nc3)=O)CCOCC2)CCCCCC1=O C(CC(C(C)(C)C)NC(C1CCCO1)=O)N(C(Cn1c(C)csc1=O)=O)C N1(C(C2CC2C(F)(F)F)=O)CCN(CCc2ccccc2Br)C(CCO)C1 CC#CCC(C(=O)NCC1CC1(F)F)NC(=O)Cc1ccc(O)cn1 C=CCC(C)N=c1[nH]c(NC2CC(O)C23CCC3)nc2c1CCCCCC2 N1(C(c2c(C)scn2)=O)CCOC(C(=O)NOCCC(C)O)C1 C1(CNC(c2c(CCC)occ2)=O)CCC(C)N(C(=O)C=Cc2ccnn2C)C1 C=CC(CC)CC(=O)N(CCCCN(C(=O)C(F)(F)c1nccn1CCC)C)C N1(C(CC2(C)CC(F)(F)C2)=O)CCC2(CC1)CCN(C(c1coc(Cl)n1)=O)CC2 N(C1c2ccccc2CC1NC(C1CC(CF)C1)=O)C(C1(C(C)C)COC1)=O CC(F)(C(=O)NCCC1CC(NC(c2ccco2)=O)C1)c1ccccc1 C1(NC(C(C2CC(F)(F)C2)OC)=O)CCCC1NC(C1CCOCC1)=O C1(NC(C2(CCC)CC2)=O)CC(NC)CN(C(=O)C(CC)N(CC)CC)C1 C(=O)(C1=CCCN(C(C23CCC(CC2)C3)=O)C1)N1CC(N(C)C)C2(C1)CC2 C1(CC)CN(C(c2cc(C(N)=O)[nH]n2)=O)CCC1NC(=O)Cn1cnccc1=O c1(C(=O)NC2(CC)CN(C(C3CCOC3C)=O)C2)cnncc1OC C(C(C(C)C(C)C)NC(c1sccc1C#N)=O)NC(c1c(CC)ccs1)=O c1(C(C)(C)OC)nc(=NC(=O)N2CCC(C3OCCO3)CC2)s[nH]1 C(=O)(C(C(CC)CC)OC)NCC(C(C(=O)NC(CC=C)CO)F)C CC(CN=c1nc(N2CCOC(C3CC3)C2)c2[nH]ccc2[nH]1)c1ccsc1 CC1C(NC(=O)C=Cc2cccc(F)c2)C(C)CCN1C(C1CCCN1C)=O C=CCC(CC)C(=O)NC1(CNC(=O)CCCSC)CCOC1 N1(C(C(C)C2CC2)=O)CCCC(CN(C(=O)C(=C2CCCCC2)F)C)C1 c1(C(N(CC(=O)NC)CC(C)(C)C)=O)ccc(C)o1.C12CN(C1)C2=O CC1CN(C(C2CCOCC2)=O)CCN1c1cc(-n2ccnc2)ncn1 Cn1ncc2c(NCCF)nc(N3CCC4CCC(C4)C3)nc12 c1(OC)cc(F)c(F)cc1NC(=O)NCCC1CCCC1(C)C CC1C(NC(c2ccc(CO)o2)=O)C(C)CCN1C(c1cccc2[nH]ncc12)=O C1(NC(COc2ccc(C(=O)NC)cc2)=O)CC(C)CN(C(=O)CCC=C(C)C)C1 c1(N(CCC(=O)NCCC#N)C)ccnc(N2CCC(OCCOC)CC2)n1 N1(C(=O)CN2CCCC2=O)CCCN(C(=O)C(C2CCOCC2)O)CC1 C12(C(=O)NC3C(CNC(C(C)(C)c4ccccc4)=O)C3)CC3CC(C(=O)N1)C2C3 c1(NC(C(N2CCCC(c3scc(C(C)(C)C)n3)C2)=O)=O)ccccc1C#N C(=O)(CCCC(CCC)CCC)NCCCCCNC(C(C=C)(C)C)=O C1(C(=O)NCC2(CNC(C3(CC)CC3(F)F)=O)CCCC2)OCC2CCCC1C2 c1(C(=O)NCC2(NC(CCNC(C3C(C)C3)=O)=O)CCOC2)cc(CO)n(C)n1 C(=O)(C1=CC(C)(C)C1)NC(c1ccccc1)C(=O)NC(C#C)CCC c1(C(N2CC(OC)(CNC(=O)CCCN(C)C)C2)=O)ncccc1C(F)(F)F C#CC1(C(=O)NCC(C)(O)C(F)F)CCN(C(=O)Cn2cc(Cl)cn2)C1 C(=O)(C#CC1(C)CCCO1)N1C2CN(C(c3ccn(C)n3)=O)C(CC2)C1 N1(C(C(CC2CC2)OC)=O)CCC(C(=O)NC2CCCC2)(OC)C1 N1(C(CC(=O)OCC)=O)CCC2CCCC12C(=O)NC(C)Cc1cccnc1 Cc1cc(C)c(C(=O)NC2CC2CNC(c2cccc(OCCF)c2)=O)cc1C N1(C(c2nc(CC)sc2)=O)CCN(C(=O)C(C)N(C)C)CC1c1cn[nH]c1 c1(C(c2n(CC)nnn2)NCC(O)CC(C)C)c(Br)cnc(Cl)c1F C1(C(N2CCC(CCC)(CO)C2)=O)CCC(C)N(C(c2cnsc2)=O)C1 C(=O)(C1CC(=O)c2c(F)cccc21)N1CC(O)(CCNC(c2cncnc2)=O)C1 N1(C(C(c2cccs2)NC(c2cc(C)oc2C)=O)=O)CC(C)C(F)(F)C1 c1(C(=O)NC2CC(NC(C(CC(C)C)N(C)C)=O)C2)cc(F)c(Br)cc1F c1(NC(CC2CCC(C(N)=O)C2)=O)cccc(S(=O)(=O)C(F)F)c1 N1(C(CCSCC(N)=O)=O)CCC(NC(=O)CCCc2cncs2)CC1 c1(C(N2CCCC2c2cc(C)no2)C(=O)NCCC)cccc(CO)n1 CC(C)C(F)(F)CC(=O)NCC(c1ccccc1)NC(=O)C(O)Cc1cn(C)cn1 C1(C(=O)NC2CC(CC(=O)OC)C2)CCCCN(C(C2(C)SCCCS2)=O)C1 C=C=CCCC(=O)N(C(C)C(=O)NCCC(C)(C)C=C)CC C(CCO)(C(F)(F)F)NC(C1(CNC(C2CC23CCOC3)=O)CCC1)=O N1(C(C(COCC)C)=O)CCC(CNC(c2ncoc2C(C)(C)C)=O)C(O)C1 N1(c2cc(C)ncn2)CC(NC(=O)CC2CCC(C)C2)C2(CCOCC2)C1 C1(O)(CNC(c2ccc(=O)n(O)c2)=O)CCN(C(C2CCSCC2)=O)CC1 N1(C(c2cccc(NC(C)=O)c2)=O)CC2CC1CN2C(=O)Cc1ccc(Br)cc1F c1(C(N(CCNC(CC2(C#N)CC2)=O)CC2CC2)=O)ccc([N+](=O)[O-])nc1 C=C=CC(C)C(=O)N(C1CCCN(C(=O)CCNC(N)=O)C1)CCO C1(C(=O)NCC2CCSC2)C2CC3C(C2NC(=O)CC(Cl)Cl)C13 C(C1=CCN(C(=O)Cc2ccnnc2O)CC1)NC(C1N(S(C)(=O)=O)CCC1)=O C1(CNC(COCc2cccc(C)c2)=O)CN(C(=O)CCCC2CC2)CCC1O C1(NC(CC(C=C)C)=O)CCCCCCC1NC(=O)C(CC)N(C)C N1(C(C2(CC=C)CCN(C(=O)C(C3CCOCC3)=O)C2)=O)CCC2C(O)CC12 c1(C(=O)NCC(C)(C)NC(=O)CNS(C)(=O)=O)cccc(C(C)(C)C(F)(F)F)c1 c1(C(=O)NC2CN(C(c3cc4n(c3)CCC4)=O)CC2O)c[nH]c2nccc(Cl)c12 CC(C)CC(C)(CO)NC(C1CC2(CC(NC(C3CCCN3C=O)=O)C2)C1)=O C(CCC(C(=O)NC1CCN2CCC1C2)NC(=O)C=CC1CCC1)OC Cn1cc(C=CC(=O)NCC2(O)CCN(C(c3cnc(C4CC4)nc3)=O)C2)nn1 CCCCCCC(F)C(=O)NCC1C=CCN1C(=O)Cc1cc(F)c(N)cc1F Cc1oc2ccccc2c1CC(=O)NCC1CCCN(C(C2CNC(=O)C2)=O)C1 N1(C(c2c(C)nc(CC)o2)=O)CC2CC1CN(C(C1CC3(CCCCC3)C1)=O)C2 C1(NC(c2ccc(OCC(C)C)cc2)=O)CCN(C(=O)CCC#N)C(C2CC2)C1 N1(C(C(C)Cc2cccc(F)c2)=O)CC2CC(CNC(=O)CCC3(C)CC3)C2C1 C12(NC(c3cc(Cl)c(Cl)nc3Cl)=O)CCCC1N(C(c1ccc(Cl)cc1)=O)CC2 CC1(C)C2CN(C(c3cc(-c4nc(-c5cccc(CO)c5)no4)ccn3)=O)CC12 N1(C(C2(OC)CCCC2)=O)CC2CC2(CNC(c2ccncc2F)=O)C1 C1(N(C(C(CC)=CC)=O)C)CCN(C(=O)CCc2ccccc2O)CC1C C12(C)CCC(C(=O)N(CC(CC)NC(=O)CCC(=O)OC)C)(CO1)C2.CCO C1(C(=O)NCC2N(C(c3ccc(C)c(C)c3)=O)CC2)CCCC2(CCC2)O1 c1(CNC(C(C)N(C(C2C3CCC(F)C23)=O)C2CC2)=O)ccc(F)cc1F c1(OC)ccc(C(N2CCC3C(NC(=O)C(C(C)(C)C)SC)C3C2)=O)c(N)c1 C1(NC(C2CCCN(CCC)C2)=O)CCCN(C(c2ccc(Cl)cn2)=O)C1C C(=O)(C(O)CC(C)C)NC1(c2ccccc2)CN(C(C(CCSC)O)=O)C1 C(=O)(C(C(C)(C)C)C1CC1)N(CCNC(c1cc(CCOC)on1)=O)C c1(OC)csc(C(N2CCCC2C(C)NC(C2CC23CC3)=O)=O)c1OC c1(NC(C2C(C(=O)Nc3c(C#N)ncc(C)n3)C2)=O)c(F)ccc([N+](=O)[O-])c1F c1(CNCC2CCCN(C(CS(N)(=O)=O)=O)C2)cc(=O)n2ccccc2n1 c1(C(C)C)cccc(C(C(=O)NCc2cccc(Cl)c2)N(CC(Cl)Cl)C(C)C)c1 O=S(=O)(CCCCCl)N1CC2CC2(CNCc2cscn2)C1 N1(C(C)=O)CC(c2nnnn2C)(NCCc2nnc(C(C)C)s2)C1 CCCCC(C)(C)NC(=O)CC1CCCCN1C(C1CCOCC1)=O C1(NC(c2on(C)c(=O)c2)=O)CCC(C)(C)CC1CNC(c1ccnnc1)=O C(=O)(CCCCC(F)F)NC(CCN(C(c1c(CC)nc(=N)[nH]c1)=O)C)C N1(C(C(CCC)C)=O)CCC(C(=O)NC(C(N)=O)C2CCCC2)CC1(C)C C1(NC(C(CC=C)CC)=O)CC2CCC(C1)N2C(C1(F)CCCC1)=O c1(OC)c(CC(N2CCCC(C)C2CCNC(=O)C(C)C)=O)cccc1Br C1(C(=O)NCC2CCN(CCC)C2)(CO)CCN(C(=O)C(C)N2CCCC2)C1 Cc1cc(=NCc2cnccc2C)[nH]c(N2CC(=O)NC(C(C)C)C2)n1 C(C(CC(C)C)C(=O)N1CC2CCC1(CNC(=O)Cc1cccs1)CC2)OC C(c1cnc(C(C)(C)C)s1)=CC(N1C(CNC(C2N(C)CC2)=O)C=CC1)=O c1(CC(=O)NC2CCCN(C(Cn3c(C)ccn3)=O)C2)c[nH]c2ncccc12 Cc1cc(C(=O)N(CCCNC(C2CSCC(=O)N2)=O)C(C)C)n(C(F)F)n1 CC1CN(C(c2c(CNC(=O)Cn3ncnn3)cnn2C)=O)CCC1CO CCC(C)(C)C(O)C(=O)NCC(C1CCC1)NC(c1cccn1C1CCCC1)=O C(=O)(C1CCCc2c[nH]nc21)NCC1(CNC(=O)Cc2cnns2)CC1(F)F C1(CNC(c2ccc(C)nc2O)=O)CN(C(C2CCOC2)=O)CC(C)(C)C1 N1(C(C(CC=CCC)C)=O)CC(C(=O)NC2CCOCC2OC)CCC1(C)C CC1C(C(N2CC(N=[N+]=[N-])C2)=O)CCCN1C(c1sccc1C#N)=O n1(CC(=O)NC(CC)CNC(=O)Cn2cc(C(C)O)nn2)cc(S(C)(=O)=O)cn1 C=CCC(C(=O)NCC1(OC)CCN(C(=O)C(C)=CCC)C1)OC CC1=C(C(=O)N2CCN(C(C3COC(=O)N3C)=O)CC2C)CCCC1 c1(C(C(=O)N(CCNC(=O)Cc2cc(C)no2)CC)=O)ccc(F)cc1 c1(C(=O)NCCOCCCNC(C2CN(C(=O)NC)C2)=O)cc2cnccc2o1 C1(C(=O)NCC2ON=C(CC)C2)CCC2(CCCCC2)CC1 n1(CC)cc(CC(N2CCCCC2CCNC(=O)CCCSC)=O)c(C)n1 N1(C(CC(C=C)C)=O)CC(C2CCCN(C(=O)Cn3ccnn3)C2)C1 c1(C(N(C2CCN(C(=O)C(CC)CC)CC2)CCC)=O)ccsc1C#N n1(CC(=O)NCC=CCNC(CN2C(C)CC2)=O)c(C(F)F)nc2ccccc12 N1(C(c2c(CCNC(C(C)=C(CC)C)=O)n[nH]c2)=O)CCOCC1C N1(C(=O)C=C(Cl)Cl)CCCC2C1CCN2C(=O)C(O)Cn1cncn1 N1(C(Cn2c(C)nnn2)=O)CC2C=CC1C(C(N1CC(O)(C3CCC3)C1)=O)C2 Cc1cc(C(=O)NCC2CC2NC(c2c(C(F)F)n[nH]c2C)=O)c(Br)s1 CC1=C(C(=O)NCC2CCCC2NC(c2cc(F)ncc2C)=O)CCC1 N1(C(C=CC(=O)NCC(=O)NC2CC2)=O)CC2(CCOC2=O)C1 C1(NC(C(CCOCC)C)=O)CN(C(=O)CSc2ccc(Cl)cc2Cl)CC(C)(C)C1 C12(NC(c3c(C)nn[nH]3)=O)CCC(CN(C(C3CCCC4(CCC4)C3)=O)C1)C2 CC1(C#CC(=O)N2CC(CNC(C3CC(=C4CCC4)C3)=O)C3(CC3)C2)CCCO1 c1(NC(=O)NC(COC)C)cc(CNC(c2ccoc2)=O)on1 C=CCCCCCCC(=O)NCc1c[nH]nc1C(=O)NC(COC)CCO Cc1ccn(C)c1C(N1CCCC(NC(=O)CC2CC(N(C)C)C2)C1)=O Cc1cc(CC(N2CCC(N(CCO)C(C3CNC(=O)N3)=O)C2)=O)cs1 C(=O)(C(C)(C)C(C)O)N1CCC(OCC(=O)N(CC=C)CCOC)C1 c1(C(=O)NC(CN(C(C2CCCCS2)=O)CC)C)sccc1C1CC1 c1(OC)nc(N2CCCC2CCCNC(C2CC3CCC2C3)=O)nc2[nH]cnc12 C1(C(N2CC(C(=O)NC)C2)=O)CC1C1CN(C(c2cccnc2)=O)C1 c1(C(N(CC(CC)NC(c2ccsn2)=O)C)=O)cccc(Cl)c1 Cc1occc(=O)c1OCC(N1CC(O)(CNC(=O)CCC(C)(C)O)C1)=O c1(C(N2CCC(CNC(=O)Cc3ccncc3Cl)C2)=O)cnc2c(c1)CCC2 C1(CNC(CNC(CC)=O)=O)CCC2(CN(C(C34CC(C(=O)OC)(C3)C4)=O)C2)O1 Nc1cccc(Cc2nc(NC(=O)NCC(c3cc(Br)cs3)O)cs2)c1 C1(=O)C(O)C(C)(C)C(=O)NC(C)CCN1.c1(C(=O)OC(C)(C)C)n[nH]cc1Cl c1(C(N(c2cccc(SCC)c2)C)=O)cccc2c1CC(C(=O)OC(C)(C)C)C2 N1(C(c2cc(CCC)on2)=O)CCC(NC(C2(C#N)CC2)=O)C(CC)C1 CC1CN(C(c2ncnc(O)c2F)=O)CC(C)N(C(c2c(F)cccc2F)=O)C1 c1(C(C(=O)NC2C(CNC(c3cc(C)sn3)=O)CCC2)O)cn(C)nc1C C1(CNC(COC(CC)C)=O)CCN(c2nccc(C)n2)CC1C C1(C(=O)NC(C)(C)CNC(c2cc(Cl)ccc2C(F)F)=O)CCc2cncn2C1 c1(C(c2nnnn2CC(F)F)NCCCOCC)c(Cl)cc(C(=O)OC)nc1Cl C1(OC)C=CCN(C(C2CC(C)CN2C(=O)C(C)OCCC(C)C)=O)C1 C1(N=[N+]=[N-])(C(=O)NCCS(CC)=O)CCN(C(=O)CCc2ccccc2)C1 N1(C(CCC2CCCN(C(C3(CCC=C)CC3)=O)C2)=O)CCC2(CCO2)C1 CC1CC(CO)CN(C(=O)C(c2ccncc2)NC(c2c[nH]c(=O)cn2)=O)C1 N1(C(CSC)=O)C(CNC(=O)C(Cc2ccsc2)NC=O)CC2CCCC12 C(=O)(C1(C)CCn2ccnc21)N1C(C2CCN(C(C(C)OC)=O)CC2)C(C)(C)C1 C1(NC(C=CCC)=O)(OC)CN(C(=O)C(C)NC(=O)NC2CCCC2)C1 C12CC3(C1C=CN3CC(=O)O)CC(CCCC(C)SC(C)(C)C)N(C)C(=O)OC2 C1(CCN(C(=O)C=Cc2ccncc2)C)CCN(C(C2(C)CC3CC3C2)=O)CC1 N1(C(CC2(OCC)CCCC2)=O)CCN(C(C2CC2CF)=O)C2COCC12 c1(C(N2CCC(CC(C)NC(C(CCC)(C)O)=O)CC2)=O)scc2c1CCCC2 C1(C(=O)NC2(C)CC(N(C(=O)COCCCN=[N+]=[N-])C)C2)CCC(C)CC1 N1(C(c2cc(OCC)no2)=O)CCC(NC(c2cnn(C)c2Cl)=O)CC1C C1(CNC(c2cscn2)=O)COCC1NC(C1CCCN1C(=O)C(F)(F)F)=O C1(NC(C(=Cc2cccs2)C)=O)CC2CC(C1)N(C(=O)Cc1ccc(Cl)cn1)C2 N1(C(c2nc(C(C)OC)sc2)=O)CCCCC1CNC(C1CCOCC1)=O C(=O)(CS(=O)(=O)C(C)(C)C)NCC1CC(OC)CN1C(c1cc(O)cs1)=O c1(C(N2C(C(C)(C)NC(C(C)CO)=O)CCC2)=O)n[nH]c2cc(Br)ccc12 N1(C(C(F)=CCC)=O)CC2CCCC2(NC(=O)Cc2cccc(C)c2)C1 c1(N(C2CCCNCC2)C(C)=O)ccc2c(c1)N(C(=O)CCC(N)C(N)=O)CCO2 C1(C(=O)NCC(C(=O)NC)C)CNC(=O)CN1C(c1n[nH]cc1C)=O C1(C)(CC(=O)NCCC(C(=O)OCC)C)CC(F)(F)CN1C(=O)OC(C)(C)C C1(N(C(=O)C(O)CNC(=O)CCc2ccc[nH]2)C)CS(=O)(=O)C1(C)C c1(NC(CN2CC(NC(C(C)(C)C(N)=O)=O)C(C#N)CC2)=O)nccc2cccnc12 N1(C(CC2(OC)CCCCC2)=O)CCCC(F)(CNC(C2(Cl)CC2(F)F)=O)C1 C1(NC(C(C)NC(c2cnnn2C2CC2)=O)=O)C2CCCC1CC2 N1(C(COCC#C)=O)CCCC(NC(C2C3(CC3)C23CC3)=O)C1 c1(OC)ccncc1C(N1CCCC1CC(=O)NC(Cn1cccn1)CO)=O c1(CC(=O)NCCC2CC(NC(CNC(C)=O)=O)C2)ccc(F)c(Br)c1 C(=O)(CCN=c1[nH]ccs1)N(CCOCCNC(C(C(=O)OCC)C1CC1)=O)C CCC(CC)CC(F)C(=O)NCC1CC1CNC(=O)C(C)(C#N)CC C1(c2cn(C)nc2)CC(C(=O)NS(=O)(=O)CCCC2CCCCC2)CCO1 C1(NCc2c(C)cccc2C)CC2CCC(C1)N2S(=O)(=O)C1CCCCC1 C(=O)(C(C)CC(C)C(C)=O)NCCC1(C(=O)NC2C(C#C)CCC2)CC1 N1(C(CNC(C(N2C(COC)C(C)(C)C2)=O)=O)C)CCc2ccccc21 c1(-n2cc(C(C)NC(C34CCC(C3)C4(C)C)=O)nn2)c(F)cccc1F c1(C(=O)NC(C)CNC(c2sccc2-n2ccnn2)=O)cnc2cnn(C)c2c1 N1(C(c2cc(COC)no2)=O)CCC2(CCN(C(c3ccc(Br)o3)=O)C2)C1 N1(CCNC(C2C(C(=O)OC)C2)=O)CCN(C(=O)CCN2CSCCSC2)CC1 C1(CN(C(C(COC)C)=O)C)C2CN(C(c3cc(C(F)F)cs3)=O)CC12 Cc1ccc(CCC(=O)N(c2cccc(Cl)c2C)CC2CC2)cc1F C1(CC(=O)NCC(C(=O)NC)(C)C)CC(C)(C)CN1C(=O)C(O)C1CCCC1 N1(C(C2CC(OC)C2)=O)CC(CNC(c2ccc(O)c(F)c2F)=O)CC12CCC2 C12(CCC=C)CN(C1)C2=O.c1(C)ocnc1C(=O)O.C1(C)(CNC(C)=O)CSC1 n1(CC(=O)NCC2CC(NC(c3snnc3C3CC3)=O)C2)cc(C2CC2)nn1 C(C(O)C(F)(F)F)N(C)CCN(CC(C(=O)OC(=O)OC(C)(C)C)CO)C(C)=O CCCS(=O)(=O)CC(=O)N1CCC(NC(=O)Cn2cccn2)C1C(C)(C)C C1(CNC(CCC(C)SC)=O)CN(C(=O)Cc2cn(C)nn2)CCN1C N1(C(c2c(CC)cco2)=O)CCC(C(C)(C)NC(c2ccoc2Cl)=O)CC1 CCCCCCNC(=O)CC1(CNC(=O)C(C)COCC)CC1 C1(C(N(CC(=C)C)C)=O)CC(F)(F)CN1C(C1C2CCC(F)C12)=O c1(-c2cn(C3CN(C(C(C)NC(COC)=O)=O)C3)nn2)cccc(C)n1 O=C1CCN(CCOc2ccc(Cl)c(Cl)c2)C(=O)N1CC1CCC2(COC2)O1 C1(NC(C2C=CCN2C(c2cnc(Cl)s2)=O)=O)CC2OCCCC12 C(C)(C)(CC(=O)N(C1CCN(C)C1)C)NC(CC1ON=C(C)C1)=O c1(C(N2CC(N(C(=O)C(C3CCCC3)c3cccs3)C)C2)=O)ccc2c(c1)COC2 C1(CC=C)(NC(c2nnn(C)n2)=O)CCN(C(C2CCCCC2C(C)(C)C)=O)C1 c1(C(N2CC(OCCNC(C(C)(C)F)=O)C2)=O)ccccc1Cn1ccnn1 N1(C(C(C)N(CC)CC)=O)C(C(N2CCC2(C(C)C)CO)=O)CCC1C(C)C Cc1cccc(CC(=O)NC(C)CNC(c2cnc(O)n2C)=O)c1 c1(C(C(=O)NC2CCN(C(CCCOC)=O)C2)(C)C)ccc([N+](=O)[O-])cc1F N1(C(c2ccc(C(C)O)cc2)=O)CC2CC(C)N(C(=O)C3=CCC3)C2C1 C1(C)(CNC(CC2(OC)CN(C(C3CCCCC3O)=O)C2)=O)CC2(CCC2)C1 N1(C(c2c(C)nc(N(C)C)s2)=O)C2CCC1CC(NC(C1(C3CC3)CC1)=O)C2 c1(OC)cnc(C(=O)NC2CC2CNC(=O)CC2CCN(C(C)=O)CC2)c(F)c1 c1(NC(CC2CN(C(C(C)=CC(C)(C)C)=O)CC2C)=O)cccc(Cl)c1 N1(C(C2C(Cl)(C(N(C)C)=O)C2)=O)CCOC(C)(C(=O)OC(C)(C)C)C1 C1(NC(=O)CCc2cnc[nH]2)C2CCC(C2)C1C(=O)NCC(c1ccccc1)O c1(OCC)cncc(C(=O)NCC(C2CCC2)NC(=O)Cc2csnc2C)c1 C(=O)(C(F)C(=O)NCCC(C)CCNC(=O)CCNC(C1CC(OC)C1)=O)OC C(=O)(CC(C(C)C)NS(=O)(=O)CCc1ccsc1)NC N1(C(CC2N(C)CC=CC2)=O)CC2(CCCC2NC(=O)CCC(N)=O)C1 c1(OC)ccc2[nH]c(=NCC(F)F)[nH]c(=NC(C)c3ccc(Br)cn3)c2c1 c1(C(CNC(c2cc(Cl)no2)=O)NC(C(F)OC)=O)ccc(F)cc1F c1(CC(N2CCCC(C)(CNC(=O)CCCF)C2)=O)csc2c(F)cccc12 CCC(C)C(C(=O)NCC#CC(F)(F)F)N(C)C(c1cc(F)cc(F)c1)=O Cc1cc(F)cc(C)c1CNC(c1nnnn1C1CC(F)(F)C1)c1nncs1 C#CC1CN(C(=O)CCc2ccc(C)o2)CCN1C(=O)Cc1ccc(CC)cc1 c1(C(=O)NC2COC3CN(C(C(N)=O)=O)CC32)cc(S(N)(=O)=O)ccc1Br C1(NC(CC=C)=O)CCS(=O)(=O)C12CN(C(=O)CCC(=O)c1ccc(O)cc1)C2 C#CC1(NC(C2CCCC2NC(=O)CC2CC=CCC2)=O)CCCOC1 N1(C(CCC(=O)OC)=O)C2CCC1CN(C(=O)CCC1CCOC1)C2 c1(CC)nc(C)oc1C(=O)N(C1CCCN(C(=O)Cc2ccccc2)C1)CCF c1(C(N2CCC(OC(F)F)C2)=O)cccc([N+](=O)[O-])c1Cl.C12CC(C(O)C1O)N2 CCC(CC1CCCCC1)C(=O)NCC1CC(F)CN1C(c1ccnc(Cl)c1)=O CCCC(O)C(=O)NCC1CC(NC(c2cc(SC(F)(F)F)c[nH]2)=O)C(O)C1 Cc1cc(C(=O)NCCC2CN(C(c3nnc4ccccn34)=O)C2)c(O)c(C)c1 c1(C(c2nnnn2CC2CC2)NCC=CCCC)cn(-c2ccccc2)nn1 c1(C(N2CC(NC(CC3(C)CC3)=O)C(N=[N+]=[N-])C2)=O)cccc2nc(O)ccc12 N1(C(C2N(C(CNCCO)=O)CCC2)=O)CC(CO)C(F)C1.NC(=O)C C1(CC=C)(NC(=O)CCCC2CCCC2)CN(C(C2CCC2C)=O)C1 C1(CC(=O)NC(C)CNC(=O)CCc2cnoc2)CCCNC(=O)C1 Nc1cc(F)c(Cl)cc1C(=O)NC1(CNC(C2CCC2)=O)CCCC1 N1(C(CCC=CC(C)C)=O)CC(CN(C)C)C1(C)C c1(C(=O)NC(C)(C)CCCNC(C2CC3(C2)CC(F)C3)=O)cnn2ccccc12 C(=O)(CS(=O)c1ccc(Cl)cc1)NC1CC(NC(C(C)(F)F)=O)CC1O c1(OC(C)(C)C(=O)NCC2CC(NC(=O)C(O)C(F)(F)F)C2)ccc(F)c(F)c1 C1(CC(=O)N(C(c2nccs2)C)C)CCCCC1NC(C1CCCCN1C)=O c1(C(=O)NC(C(C)C)(C)CNC(=O)C(C)S(N)(=O)=O)ccc2ccnn2c1 CCCC(C)(O)CC(=O)N1CC(CNC(=O)Cc2ccns2)(COC)C1 C12(c3cn(CCOCCNC(CC4(COC)CCCC4)=O)nn3)CCC(CC1)C2 Cc1ccc(C=CC(=O)NC23CC(NC(=O)COc4cnn(C)c4)(C2)C3)nc1 N1(C(C2(n3cc(Br)nn3)CC2)=O)CCCC1C1CCOCC1 N1(C(c2c(CNC(CCC#C)=O)nccc2)=O)CC(=O)NCC1C N12CCCCC13CN(C3)C(=O)c1cc(oc1)C2=O.c1(OCC(=O)O)ccsn1 N1(C(CC(C)SC)=O)CC(NC(c2cnc(SC)nc2O)=O)CC(F)C1 c1(OC)cccc(COC(C2CCC(c3ccccc3)N2)=O)c1 c1(CNC(c2ccc(C3CC3)cc2)=O)ccc(NC(C2(COC)CC2)=O)cn1 C1(CN(C(C(C)=C2CC2)=O)C)CCN(C(=O)CCc2n[nH]c(=N)s2)C1 C=CC(CC)CC(=O)N(C)CC1CCN(C(C2(n3cccc3)CCCC2)=O)C1 C1(C(N(CCOCCN(C(C(CC)C#N)=O)C)C)=O)Cc2c[nH]cc2S1(=O)=O c1(OCC(=O)NC(C)C)ccc(-c2noc(C(C)C(O)C(C)C)n2)c(Cl)c1 N1(C(C(C)=CC)=O)CCC(CN(C)C(c2cnc(C(=O)OC)s2)=O)C1 N1(C(CC2N(C(c3cc(C)nnc3C)=O)CC(C)(C)C2)=O)Cc2cnn(C)c2C1 c1(NC)c(C(=O)NCCNC(C2(COC)CCOC2)=O)cccc1F c1(C(=O)NCC2(CNC(C3C(C)C3)=O)CC2)csc2cc(Cl)ccc12 c1(C(=O)NC2CN(C(c3ncc(OC)cn3)=O)CC2F)cc(SC)ccc1OC C12(NC(CSc3cccc(OC)c3)=O)CCCN(C(=O)CCOC(C)=O)CC1C2 c1(C2(NC(C(CC)c3ccccc3)=O)CC2)ccc(O)c(F)c1 c1(CC)cc(CNC(c2nnnn2C2CC(CC)C2)CC2CCOC2)ccn1 N1(C(c2cnn(CC)c2C)=O)CCC12CN(C(c1cc(=O)c(O)c[nH]1)=O)C2 C1(C(=O)NC(c2cccnc2)C(=O)N2CCC2C2CCCC2)CC=CC(O)C1 c1(C(N2CCCN(C(CSCCOC)=O)CC2C)=O)cc2ccccc2cn1 N1(C(C(CN(C(CCSC)=O)C)C)=O)CCCC[Si](C)(C)C1 c1(CC(=O)N(CC(CC)NC(=O)C(F)Cc2ccccc2)C)ccc(O)nc1 C(=O)(C(CCSC)OCC)N1CCCC1C(=O)Nc1ncc(C(=O)OCC)o1 Cc1nn(C)c2c1NC1=NC3CC(C3)NC2=N1.C1CCCCCCC1 c1(CC(n2cc(CN(C(C(C=C)OC)=O)CC=C)nn2)C(=O)O)ccc(Cl)cc1 c1(C(N2CC3C(C(=O)NC(CC)C(N)=O)(C3)C2)=O)ccc(C(F)(F)F)c([N+](=O)[O-])c1 C(CN=C(NCC1COC(C)(C)O1)N1CCCCCCCCC1)SC Cc1ncc(C(N2CCC(CO)C(NC(c3cnn(C)c3F)=O)C2)=O)c(C)n1 C1(OCCC)CCCN(C(c2cnn(CC)c2)C(=O)NCC(C)C)C1 CS(=O)(=O)c1ccc(C(N2CC3CC2CS3)C(=O)NCc2ccccc2Br)o1 C1(CC(=O)NCCOC(C)=O)CN(C(=O)CCC2CCCCC2)C(C)(C)C1 n1(CC)ncnc1C(C)NC(C1(CNC(C2(C)CCCC2)=O)CC1)=O N1(C(c2c(OC)oc(C)n2)=O)CCN(C(C2CC2C(F)F)=O)C(C)C1 Cc1cc(NC(C2(O)CCN(Cc3cc(C)n(C)n3)C2)=O)cc(Br)c1C Cn1ccnc1C(=O)NCCc1ocnc1CNC(C1CCC1F)=O C(=O)(C(CC)C(C)C)N1CCC(CC#C)(C(=O)NCc2conc2C)C1 c1(OC)nccc(C(=O)NC2CCCCN(C(=O)C(c3ccc(Cl)s3)=O)C2)c1Cl C(CC1=CCN(C(=O)C(F)CC2CCC2)CC1)NC(C1Cc2nccnc2C1)=O N1(C(c2c(CC)[nH]cc2)=O)CCOCCC1C(=O)NCCn1nncc1C C(C1=CCN(C(=O)Cc2ccnc(Cl)c2F)CC1)NC(C1C(C(C)O)C1)=O C1(C)(CNC(C2(C)CCCCC2)=O)CCCN(C(=O)C=Cc2cscn2)C1 C=Cc1cncc(C(=O)NC2CC3CCC2(CNC(c2ccnc(O)c2)=O)C3)c1 C1(OC)CC2(C1)CC(C(=O)NCCC1CCN(C(=O)C(C)=C3CCC3)C(C)C1)C2 C1(C(=O)Nc2c(C)cc(Cl)nc2)CC(O)C(N=[N+]=[N-])C1 C=C(C)C(O)CC(=O)NCCNC(c1cccnc1N)=O c1(C(c2cn[nH]c2)NC(c2ccco2)C)nnnn1CCC1CC1 N1(C(C(C)(C)OC(C)=O)=O)CCCC(CO)(NC(c2ccc(C(N)=O)cn2)=O)C1 c1(NC(=O)NCC(C)OC)cc(CN(C)C)cc(F)c1 c1(C(=O)NCC2CC(NC(C(C3CCCOC3)OC)=O)C2)cccc(C#N)c1 c1(CCC(=O)NCC(C)(CC)NC(C(COCC)C)=O)ccc2c(c1)COCC2 C1(F)(CNC(C(c2ccc(Cl)s2)C)=O)CCN(C(C2CCCN2C=O)=O)CC1 N1(C(C(C)OCCC=C)=O)CC(C)(C)C(NC(=O)CN2CC3CC3C2)C(C)(C)C1 C1(NC(C(C)OCC(F)(F)F)=O)CCCCC1CNC(=O)CC1CC(C)(C)C1 Cc1csc(Cl)c1C(=O)NC1CC1NC(=O)C(C)(C)c1ccsc1 C1(C(NOCC=C)=O)CCN(C(=O)C(C)CC(F)F)C(C)(C)C1 N1(C(CCCCCC=C)=O)CCC2(CCC(NC(=O)C(C)C=C)C2)C1 C(=O)(C1Cc2ccc(F)cc21)NC1(C2CCN(C(CCNC(N)=O)=O)C2)CC1 c1(C(=O)NCC(=O)NCC2C(C)C2)cc(C(F)(F)F)cc([N+](=O)[O-])c1 N1(C(c2n(CCC)ccc2)=O)CC(N(C)C(C2CC23CCCC3)=O)C2(CC2)C1 CCCC(CNC(c1cnn[nH]1)=O)C(=O)NCCCC1CC1 Cc1ccc(C=CC(=O)NC(C)CN(C)C(c2cc(C)c(Cl)s2)=O)cn1 c1(C(=O)NCC2CCN(C(CC(=O)OC)=O)C2)ccc(S(=O)(=O)C(F)F)cc1 c1(CCC(=O)NCC2CCCN(C(c3c(C)ncs3)=O)C2)ccc([N+](=O)[O-])cc1 c1(C(N2C(C(=O)NC3CCN(C(C)=O)C3)C=CC2)=O)cnc(O)c(F)c1 c1(C(C)C)ccc(C=CCC(=O)NCC=CCNC(C2(C)CC=CC2)=O)cc1 N1(C(COC)=O)CCCC(NC(=O)C=Cc2nnc(C(C)C)o2)C(F)C1 c1(C(N(CCC(C)NC(COCCC=C)=O)C)=O)ccc(OC(F)(F)Cl)cc1 N1(C(C2C(C=C)OCC2)=O)CCCN(C(=O)Cn2cc(C(C)=O)nn2)CC1C c1(C(N2CCC(CNC(c3ccncc3Br)=O)C2)=O)cc(F)c(F)cc1Br C1(C(=O)NCC(C)CNC(C2CN(C3CCC3)C2)=O)CCN(S(C)(=O)=O)CC1 C(CC(C)C)(C(=O)N1CCOC(COCC)CC1)c1n(CC)nc(-c2ccsc2)n1 CC1CC2CN(C(C3COCCN3C(=O)C=Cc3cccnc3)=O)CCN2C1 C1(C(=O)NC2CC(NC(CCCC(=O)OCC)=O)C2)Cc2c[nH]cc2S1(=O)=O c1(N2CCC(C(N3CCC3CNCc3cccnn3)=O)C2)ccccc1Cl c1(C(=O)NCc2ncc(C(=O)NCCC3CCN(C)C3)cn2)cc(F)cc(F)c1 CC(C)CCCCC(=O)NCCN1CCCN(C(C23CCOC2C3)=O)CC1 C1(C(N2CCN(c3ncc(C(C)=O)cc3C)CC2)=O)CCc2nc[nH]c2C1 N1(C(C2CCC(C(=O)OC)CC2)=O)CCC(NC(=O)CCCC(N)=O)C(F)C1 C1(NC(=O)NCC(CSC)OC)CCC2(CC2)C1 Cc1ccc(F)c(C(=O)NC2CN(C(=O)CSc3ccccc3O)CCC2C)c1 C1(C(=O)NC(CC2CCCC2)CO)CC1C1CN(C(=O)Cc2cscn2)C1 N1(C(=O)Nc2c(C3(C)CCO3)nccc2)CCC2(CC1)OCCO2 c1(NC)cc(Cl)ccc1C(N1CC(NC(=O)CC2CCSCC2)C2CC12)=O C1(CC(=O)NCC(C)N(C(c2cn(C(C)C)nc2)=O)C)CCN(CCF)CC1 C(CCS(N)(=O)=O)(C(=O)O)n1cc(-c2ccc(OC)nn2)nn1 C(=O)(C(F)CCC(C)(C)C)NCC1C(NC(C(C)(C)OCCC)=O)C1 N1(C(CCC2CCCN(C(=O)CCn3ccnc3)C2)=O)CC2COCC(C2)C1 C1(NC(CC2CN(C(c3c(CC)occ3C)=O)CC2C)=O)CC12CCOCC2 Cc1cc(Cl)c(C(=O)NC2CC(CNC(C3CCO3)=O)C2)c(Br)c1 C1(NC(C2N(C)CCC2)=O)COC2CN(C(=O)C=CCF)CC12 C#CCC(C(=O)N1CCC(CN(C(=O)CCn2c(C)csc2=O)C)C1)C1CC1 N1(C(CC2C(C)C(=O)CC2)=O)CC(C)N(C(c2ncn3c2CCC3)=O)C(C)C1 C=C(Cl)CCC(=O)NC1CCCC(NC(=O)C(C(C)C)N2CCCS2(=O)=O)C1 c1(C(=O)NC2CN(C(C(c3c(C)noc3C)C)=O)CC2C)noc2ccccc12 c1(C(=O)NC2CC(CCNC(C3CC(O)C3)=O)C2)cc(F)ccc1O CCCCC(C(=O)NC1CC(C)(NC(c2[nH]nnc2C)=O)C1)C(C)C N1(C(c2cc(-c3cccc(C(=O)OCC)c3)on2)=O)CCC=C(c2ccco2)C1 c1(C(=O)NC2C(NC(CC(C)c3ccncc3)=O)CCC2)nc2c([nH]1)CCCC2 C1(C(=O)O)COCCN(C(C2CCC(F)(F)CC2)=O)C1 c1(C(=O)NC(C(C)NC(CC2C(CC)C2(F)F)=O)CO)ccnn2ccnc12 c1(C(N2C(CCCNC(C(=O)N(C)C)=O)CCCC2)=O)nc2ncccn2n1 c1(C(C)C)cccc(C(=O)NCC2(C)CCN(C(=O)CC3CC3C)C2)n1 C(=O)(CC(C)CF)NCc1c(CCNC(C=C(C)C(C)(C)C)=O)ocn1 c1(NC)cc(C(=O)NCC(C)N(C(=O)C=CSc2ccccc2)C)cc(Cl)n1 c1(CC)noc2nc(-c3ccco3)cc(C(=O)NNC(=O)CSC3CCCC3)c12 C1(CC)CN(C(C2CC(C)CN2C(c2cnc(C)nc2)=O)=O)CCO1 N1(C(C(C)=NOCC#N)=O)CC(C(=O)NC2C(O)C3CCOC23)OC(C)C1 C(CS(=O)(=O)Nc1ncc(C(C2CCCOC2)=O)s1)(C1CCOCC1)OCC C(CCC(C(=O)NC1(c2nc[nH]n2)CC1)NC(=O)CCCCC#N)OC C(=O)(C(C)C(C)(C)C)N(C(C)CN(C)C(c1ccc(COC(C)(C)C)o1)=O)C C(C(C(=O)N1CC(Oc2ncccn2)C1)NC(C1CCC1C#N)=O)OCC C1(NC(c2[nH]cc(CC)c2)=O)CN(c2cc(C(F)(F)F)ncn2)C2CCCCC12 c1(OC)ccc(NC(=O)CN(CC(C)C)C(=O)Cn2cc(Cl)cn2)cc1 N1(C(C(C(C)O)NC(=O)CC2=CCCC2)=O)CCC2(CC=CCO2)C1 c12cccc(c1)C(=O)NC(CC)CNC(=O)C1CCC1C2=O.c1(S)nncn1C c1(CC)c(C(N2CCOC(CCNC(c3conc3C(C)C)=O)C2)=O)ccn1C C1(NC(CC2CCC(C)C2)=O)CCC(F)(F)C1O C1(C(=O)NC2C(CNC(c3n(CC)cc(Cl)c3)=O)CCCC2)C(F)(F)C12CCC2 C(C)(C)(C(C)CC(=O)NCc1ccc(C)o1)NC(c1c(CC)noc1)=O CCCCCCCCC(=O)NC1CC2CCC1(C(=O)NCCCCN=[N+]=[N-])C2 CCCC(CC(C)C)C(=O)NC1(COC)CCN(C(=O)C=Cc2cn[nH]c2)CC1 C1(C(=O)NCC=CCNC(CNS(CC)(=O)=O)=O)CCCCN1C c1(NC)c(C(N2CCC(C)N(C(=O)C=CC(C)(C)SC)CC2)=O)sc2nccnc12 CC(C)C(C)(CNC(=O)CCc1ccnn1C)NC(=O)CCC1CCCC(O)C1 c1(C2CCN(C(N(C(C3OCC(C)C3)=O)C)=O)CC2)ccc(Br)cc1Cl N1(C(c2c(CC)nns2)=O)CC(C(N2CC(NC(N)=O)C2)=O)CC1(C)C C(c1ccc(C#N)cc1)=CC(=O)NC(CC)(C)CNC(C1CC(C(C)C)=NO1)=O Cc1ccc(N)c(C(N2CC(C)(NC(=O)Cn3cc[n+](C)c3)C2)=O)c1 C1(C(=O)NC2C(C)(C)CN(C(=O)C(F)n3cccn3)C2)CCCCC1C1CC1 C(c1ccc(C)s1)=CC(=O)NCCN(C(c1cc(C)no1)=O)CC c1(C(=O)NC(C2CCOC2)CNC(C2CC(O)C2)=O)cc2n(n1)CCCN2 N1(C(C2(COC)C=CCC2)=O)CC2CCC(C1)C2NC(=O)C1=CCCCC1 c1(C(=O)NC2CC(C)N(C(=O)CC3CCC(F)(F)C3)CC2)ccnc2[nH]nnc12 C1(C2CCCN(C(C3CCCN3S(C)(=O)=O)=O)C2)(NC(C(C)OC)=O)CC1 N1(C(C)C)CCCC(CNC(=O)C(=O)Nc2cc(C3CC3)n(C)n2)C1 c1(C(=O)NC(C2CCN(C(=O)CC3=CCCCC3)C2)(C)C)ccc2c(c1)OCO2 CC(C)CC(C)CNC(=O)C(C)(CO)NC(=O)C(C)Cn1cccn1 c1(NC)snc(C)c1C(N1CCC1CNC(=O)C(CCSC)NC(C)=O)=O c1(C(N2C(CNC(c3ncc[nH]3)=O)CC(F)(F)C2)=O)ccc2c(n1)CCCN2 C1(CNC(C(C(C)C)N(C)C)=O)CN(C(c2nnn(C)c2N)=O)CCC1(C)C c1(C(=O)NC(CC=C)CNC(c2conc2C(C)(C)C)=O)cc(C)c(Cl)c(C)c1 c1(C(CNC(COCC(=C)C)=O)NC(=O)C(O)CN(C)C)ccc(N(C)C)cc1 c1(C(=O)NCC2CC(NC(C(c3ccccc3)OC)=O)C2)nc(C2CC2)oc1C Cc1c(C(=O)NC23CCCC2CN(C(=O)C(C)(F)F)C3)cccc1S(N)(=O)=O N1(C(CCC(C)C)=O)CCN2C(=O)C(NC(=O)COCCF)CC2C1 C(=O)(C=CS(F)(F)(F)(F)F)N1C(CCNC(c2ccc(C#N)cc2)=O)CCCC1 N1(C(NOCC=C)=O)CCC(NCC(=O)NS(C)(=O)=O)CC1 C1(C(N(C(C2CCCC2)C)C)=O)CC2(CCN1C(=O)C(=O)C1CCCC1)CC2 c1(C(=O)NCC(C)NC(CC(CC)C(F)F)=O)cc2cccnc2cn1 C(CNC(=O)C(F)OC)(CC(F)(F)F)CNC(Cc1cccc(OCCC)c1)=O c1(-c2c(CO)cc(C(=O)NCc3c(C)nn(C)c3C)nc2)ccc2cncn2c1 CCCC(CCC)S(=O)(=O)CC1CC(F)(F)CO1 c1(CC)c(C(=O)NCCC2CCCN2C(=O)CCC=CBr)cccc1C C1(N(C(c2cccc(SCCCC)c2)=O)C)CCCCN(C(=O)CSC(C)C)C1 C12(NC(CC(=C=C)C)=O)CCOCC1CN(C(=O)COCC1CCCOC1)C2 CC(CN=c1[nH]c(N2CCc3ncncc3C2)nc2c1CSC2)C(C)(C)C CC1CN(C)C(=O)CN1C(C1CCCC1CNC(=O)CC=Cc1ccccc1)=O c1(C(=O)NC(=O)OC)ccc(NCCN2CCCCC2C)c([N+](=O)[O-])c1 C(C(=O)N(CCCNC(c1cc(C)n(-c2cccc(F)c2)n1)=O)C)(C(C)C)OC c1(C(N2CCC(CNC(C(CC#C)C3CC3)=O)C2)=O)ccc2nccn2c1 c1(OC)cc(C(C)NCc2ccnn2C2CC2(F)F)c(F)cc1F c1(C(=O)NC(CSC)(C)C(=O)N(C2(C3CC3)CC2)C)cc(C)nnc1C CCS(=O)(=O)CCNC(C1(F)CCN(C(=O)C(F)CC2CCOC2)C1)=O N1(C(CNC(CCCNC(=O)OC)=O)=O)CCC(NC2CCN(C(C)=O)C2)CC1 C1(CNC(C(COC)(F)F)=O)CC2CCCCC2N1C(=O)Cc1sc(O)nc1O c1(OC)ccc2[nH]cc(CC(N3CC4(CCC4NC(=O)CC4CCC4)C3)=O)c2c1 C1(C(=O)NC2(C(=O)N(CC(O)C3CCC3)C)C(C)C2)CCC(C)(O)CC1 c1(CC(=O)N(CC(C)CNC(C2(CF)CC2)=O)C)ccnc(C(F)(F)F)c1 C1(C(=O)NCCC2CCN(C(C3CCN(C)C3)=O)C2)(COC)CCCC1 Cc1ccc(CN(C2CCCCC2c2ccccc2)C)c(Br)n1 CC(C)C(C(=O)NCC1CN(C(=O)CSC(C)C)CCO1)NC=O c12cc(nn1C)COCCCNC2=O.C1(C(N(C)CC2CCC2)=O)CS(=O)(=O)C1 C(C1=CCCCCCC1)(c1nnnn1C)NCc1cnc(C)n1-c1ccccc1 CCCC(CC)C(=O)N1CCC(O)(CCNC(=O)CCc2cnc(C)s2)CC1 c1(C(N2C(COC)CCOCC2)C(=O)NCC(C)C)ccc2ccc(Br)cc2n1 C1(=CCNC(CC=C=C)=O)CCN(C(=O)CSCC2CCCO2)CC1 C1(NC(C2(C)COC2)=O)CN(C(C2(c3ccc(Cl)c(Cl)c3)CC2)=O)CC12COC2 C1(C(C)C)C(NC(=O)Cc2ccnnc2O)CCN1C(C1CCCO1)=O c1(OC)cccc(C(F)F)c1C(N1CCC(C(=O)O)C(c2ccccc2)C1)=O C(c1ccc(F)c(C)c1)=CC(=O)NCC1N(C(COCC#C)=O)CC(O)C1 Cc1c(CC(=O)NC2CN(C(c3ccc(F)s3)=O)C2)cccc1[N+](=O)[O-] C1(C(=O)N(C2CCCC2)C)(CC)CCN(C(C2CC2(C)C)=O)C1 C(CCCC(=O)N(C)CCNC(c1ccc(-n2cnnc2)cc1)=O)SC c1(CC)cc(C(=O)NC2CC(CCNC(=O)C(C(C)C)NC(N)=O)C2)cc(F)c1 c1(C(=O)NC(CNC(c2cscc2C2CC2)=O)C2CC2)cc[nH]c2nccc1-2 C1(NC(c2n(C)cnc2)=O)CCSC12CN(C(C1CCCC13CCC3)=O)C2 C1(NCC)CN(C(=O)CC2(C)CCOCC2)CCN1C(c1cn(C)nc1OC)=O C1(CC)CN(C(=O)CCC2CCCCN2C)CCN1C(c1sc(C)cc1OC)=O C1(NC(c2cnc(CC)[nH]2)=O)CCN(C(=O)CCN2CCCCC2=O)CC1F C1(CNC(C(CC)C)=O)CC2CC2N1C(c1cccc(COC)c1)=O c1(CC)cnoc1C(=O)NC(C)C(=O)NCCCC(=O)OC c1(C(=O)NC2C=CCN(C(c3cccc(O)n3)=O)C2)c(F)cc(F)cc1Cl C1(CNC(c2c(OCC)n[nH]c2)=O)CC2CCC1N(C(=O)Cc1ncoc1C)C2 C1(NC(C(C=C)O)=O)COC2(C1)CN(C(=O)C(C)(C)c1cccnc1)C2 N1(C(C(N2CC(C(=O)O)CC(C)C2)=O)=O)CC2(C1)CS(=O)(=O)C2 c1(CNC(CCOC)=O)ccc(F)c(NS(C)(=O)=O)c1F c1(C(=O)NC2CC(NC(=O)CCC3CC3)C23CCC3)cc2c(Cl)cccn2n1 C(=O)(CCC(C)OCC)NCCC(=C)CNC(=O)CC1CCCC1O Cc1nn(C)cc1S(=O)(=O)NC1CC(C(=O)Nc2ncc(Cl)cc2I)C1 C1(N(C)C)CCCN(CC(=O)NCC2(F)CCN(C(=O)CC3CC(CF)C3)C2)C1 c1(OC)cc(C(N2CC3CC2C3NC(=O)Cc2cc[nH]n2)=O)ccc1Br C1(CC=C)(NC(=O)CC2CCCOC2)CN(C(=O)C(=O)NCC(F)F)C1 c1(C(N2CC(C(=O)Nc3c(C)ccc(F)c3)OCC2)=O)cc(C)c2cc[nH]c2c1 C12(CNC(COCc3c(C)ncs3)=O)CCC1CN(C(C1CC(F)(CO)C1)=O)C2 c1(OCC(N2C(CC(=O)Nc3ccco3)CCC2)=O)ccc2nn[nH]c2c1 C1(C(=O)OCC(=O)N(CC)CC)(COCC)CCOCC1 c1(C(N2C(C)CCC(NC(c3c(C)cns3)=O)C2)=O)ccc2cnnn2c1 C(C(=O)N=c1cc[nH][nH]1)(C1CCCCC1)OC(c1cnc(CC(C)C)s1)=O c1(C(N2C3C(NC(CC4C(C)(C)C4)=O)CC(C3)C2)=O)ccc(O)c([N+](=O)[O-])c1 CC1CC(c2nnnn2C)(NCCCOc2ccccc2)CN1C c1(N2C(Cn3cc(-c4ncc(C)cn4)nn3)CC2)nnc(O)c2ccccc12 C(=O)(C(C)C(O)CCCC)N1CCN(CC(N2CCC(C#C)C2)=O)CC1 CC1(C)C(=O)CC1C(=O)NCC1CC(NC(c2ccccc2Cl)=O)CCO1 N1(C(C=C(CC)CC)=O)CCC(CNC(=O)CCCOC)C12CC2 c1(OC)cc(C)ccc1NC(=O)NC1CCN(C(C2CCC3(CC3)C2)=O)C1 c1(C(N(C2CCN(C(=O)CCCn3cccn3)CC2)C)=O)cnn2c1SCC2 CC1CC(C(=O)N(CCC(=O)N(C)Cc2ncn(C)n2)C)CO1 c1(CC#N)n[nH]c2c1CCN(C(c1ccc(C#N)s1)C(=O)NCC(F)F)C2 C(=O)(CC1=CCOCC1)N1CCN(C(Cn2nnc(C(C)(C)C)n2)=O)C(CO)C1 C1(NC(CNS(NC)(=O)=O)=O)CCC(NC(C)(CC)c2nn[nH]n2)CC1 c1(C(=O)NCC(CN(C)C(C2(O)CCC2)=O)O)cccn1C1CCCC1 C1(NC(C=COCC)=O)CC2CC(NC(C3CCC4(CCC4)O3)=O)C1C2 C1(C(N2CCC2C2CCC2)=O)CCCCCN1C(c1ccsc1)=O CCC(CC(=O)NC1CCCC1CN(C)C(C1CCCN(C(C)=O)C1)=O)C(F)F C1(C(=O)NC(C(CO)NC(CC)=O)C)CC(=O)N(c2cccc(Br)c2)C1 N1(C(c2csc3ccccc23)=O)CCCC2(CCN(C(C3CCC(O)C3)=O)C2)C1 C1(CNC(C=CCC2(NC(Cn3ncc(CC)c3)=O)CCC2)=O)CC2(CC2)CO1 Cc1cc(CCNC(C2CCC(C)N2C(C2(Br)CCC2)=O)=O)cc(C)c1 Cc1onc(C(N2CC(NC(C3CCC=CCCC3)=O)C(O)C2)=O)c1[N+](=O)[O-] CC(C)C(C(=O)NC1CCC(NC(=O)C(C)(C)CN(C)C)CC1)N(C)C C(=O)(C(C(C)(C)C)OC(=O)CO)N(CC(C)NC(=O)CNC(=O)CCCCO)C N1(C(COC2CN(C(C)=O)C2)=O)C(CNC(=O)CC2CC2(C)C)CC2CC12 N1(C(C2C(C(=C)C)OCC2)=O)CCCN(C(C2CCC(F)(F)C2)=O)CCC1 c1(C(N2CCC(C(=O)Nc3cn(CC)nn3)C(O)C2)=O)ccc(Br)cc1C#N N#CC1(C(=O)OCCSC2CC(F)C2)CC1 N1(C(COC)=O)CCC(C(=O)NCC(C)C(F)F)(CF)C1 C1(NC(c2cc(CC)ncn2)=O)CC2CC1N(C(C1CC1c1ccncc1)=O)C2 CCC(CC(=O)N1CCCC(CCC(=O)NC(c2c(C)n[nH]c2C)C)C1)C(F)F c1(C(=O)NCC2(C(=O)OC)CC2)ccc(O)cc1N(C)C.C12CC1NC2=O C(=O)(C(C)(C)CCCF)N1CC(C)C(C(=O)NCC2CCCCC2)CC1 C1(NC(C2C(C)CCOC2)=O)CC=C(C(=O)NCc2nc(CO)n[nH]2)C1 N1(C(C=C(CCC)C)=O)CC(C)(C)CC1CNC(C1(C#N)CCCOC1)=O C1(C)(NC(CCC=C(C)C)=O)CCN(C(=O)Cn2nc(O)ccc2=O)CC1 C(=O)(CCCC(F)(F)CO)N1C(CNC(=O)CC2CCCCCC2)CC2(CC2)C1 N1(C(C(CC)COC)=O)CC(C)(C)OC2(C1)CN(C(C1(Cl)C3CCC(=O)C13)=O)C2 Cc1ccc(F)c2c1CCN(C(=O)NNC(=O)c1csc(C(=O)N(C)C3CC3)n1)C2 c1(C2C(OC)CC2)cn(CC2CCCN2C(=O)COc2ccccc2)nn1.C1(C)CC1 c1(NC(=O)NC2(c3c(Cl)cccc3Cl)CC2)cc2cccc(Br)c2[nH]1 Cc1sccc1C(=O)NCCc1cn(Cc2occc2C(=O)O)nn1 Cc1c(C(=O)NCC(C)NC(=O)CC(C)NC(N)=O)[nH]c2c(Cl)cccc12 c1(C(C(N2CC(COC)(NC(=O)CC(C)CF)C2)=O)O)ccc(OC)cc1 Nc1ccc(C(=O)NCC=CCNC(c2cn(C3CCC3)nn2)=O)nc1N C1(C(=O)NCCN(C(=O)C(C)n2cncn2)CCOC)CCCCC1O N1(C(CC(C)CNC(c2cncc(O)c2)=O)=O)CC(C)C(N=[N+]=[N-])C1 n1(CC(=O)NCC(CC(C)C)NC(c2nnc(CC)s2)=O)nnc2ccccc12 Cc1ccc(CC(C)C(=O)NCC#CCNC(=O)CSC(C)(C)C)cc1 C1(CNC(=O)CC2CC3CCC2C3)(CO)CCN(C(C2CC(O)C2)=O)C1 N1(C(C(Cc2c(C)nc[nH]2)O)=O)CCCCC1CNC(=O)C=CSc1nc[nH]n1 c1(C(=O)NCCNC(C2CC(N(C)CC)C2)=O)cnc(S)[nH]1 C(CCC(=O)NC1CCC(CCNC(=O)Cc2ccsn2)C1)OC c1(NCCCCNC(c2c(C)nco2)=O)ncccc1C#N Cc1nc(C2CC2)ncc1C(=O)NC1CCCN(C(=O)C(C2(O)CCCC2)F)C1 C(=O)(N=c1[nH]sc2ncccc12)C1(C)N(C(c2c(F)ccc(OC)c2Cl)=O)CC1 c1(C(=O)NC(CNC(CCc2ccc(C)s2)=O)C2CCC2)cc(C#N)cn1C Cc1ncn(O)c1C(N1CCC(OCC2CCN(C(=O)C3CC3)CC2)C1)=O N1(C(c2nc(C)sc2C)=O)CCCC2CCN(C(=O)CCNS(C)(=O)=O)CC12 C1(C(=O)NCC(=O)NCC=C)CC12CCN(C(c1ocnc1C)=O)C2 N1(C(c2nccs2)C)CCC(O)C(C(=O)NCCn2ccccc2=O)C1 N(C(=NCCc1cccs1)NCc1cccc(F)n1)CC(C)C#N C(CCC(C)C(=O)NCC12CC(CN1C(C1(CO)CC1(F)F)=O)C2)OC C(C)(CCCCNC(=O)C(C1(O)CCCC1)F)NC(c1c(CC)nc[nH]1)=O c1(C(CNC(C(F)=CC)=O)NC(c2scnc2Cl)=O)ccc(F)cc1F C(C(=O)NNC(=O)Cc1nccn1Cc1ccccc1)n1ncc(C)c1 C1(CNC(C2(C)CC(=C)C2)=O)CC(F)CN1C(=O)Cc1ccc(OCCC)cc1 CCC(C)(CC)C(=O)N1C2CCC(C2)C1C(N1CC2CC1CS2)=O c1(CCNC(CNC=O)=O)ccc(N2CCN(C(C3CC3C3CC3)=O)CC2)cc1 C(=O)(CC(CN(C)C)C(F)(F)F)NC(CCOC)CNC(=O)Cc1nccn1C CC1CN(c2cc(NCC34CC(CC3NC(=O)OC(C)(C)C)C4)ncn2)CCCO1 CC1CC(NC(c2ccncc2C(F)(F)F)=O)c2nccn21 c1(OC)cc(C(N2CCC(NC(c3c(OC)cccc3Br)=O)C2)=O)ccc1Br C(=O)(CC(C)=C(C)C)N(CCN(C(=O)CSC1CC1)CC)Cc1cccs1 c1(CONC(=O)C2(CCC)CC2)cccc(NC(CC(C)C(=O)N(C)C)=O)n1 N#Cc1c[nH]cnc1=NCC1CC(NC(=O)C2=CS(=O)CCC2)C1 c1(-c2cc(C)c(=N)[nH]c2)cnc2c(C(=O)Nc3cccn4cncc34)cccn12 CC1CN(CCO)CCC1N=c1ccc(Br)c(S(=O)(=O)N2CSCCSC2)[nH]1 N1(C(C2N(CC)CCC2)=O)CC2(C1)CN(C(c1nn(C)c(C)c1Cl)=O)CC2CO C1(CC#C)CCCCN1C(=O)COCCNC(=O)COCC(=C)C Cc1cc(C)c(C(=O)NC2CCCC(NC(c3cnn(C(F)(F)F)c3)=O)C2)cn1 Cc1ncnc(O)c1CCC(=O)NCCCC(C)(C)NC(c1cnsc1)=O c1(OC)cccc(Cl)c1C(=O)NCC1C(C)CCN1C(=O)Cn1nnc(C2CC2)n1 Cc1nc(CCC(=O)NCCC2CN(C(C3COC(=O)N3)=O)CCO2)oc1C N1(C(C(CSC)C)=O)CCCC2CN(C(=O)Cc3c[nH]c4cnccc34)CCC12 N1(C(C=C2CCC(C)C2)=O)CCN(C(=O)C(c2cnn(C)c2)=O)CC(O)C1 c1(C(=O)NCC2(NC(C(C)C3CCC3)=O)CCOC2)noc2c1CCCC2 c1(NC(C2CCCN2C(c2cc(Cl)n[nH]2)=O)=O)ccc(O)nc1 N1(C(C(C)CN(C(=O)CSCCC#N)C)=O)CC2COC(=O)C2C1 N1(C(c2ccc(OCC)nc2)=O)CC2(CCC2)CC1CNC(=O)C(C)S(C)(=O)=O c1cccc(Cl)c1C.Cc1ncc(NC(C2CCN2C(=O)C(=O)N(C)C)=O)n1CCl c1(C(N2CCN(C(CC3CCC(=O)N3)=O)C(CO)C2)=O)cnc2c(c1)CCOC2 C12(C(NOCCCN(C)C)=O)CC(CN(C(c3cc(F)ccc3O)=O)C1)C2 CC1(CNC(C2CC2[N+](=O)[O-])=O)CCN(C(c2coc(C3CCCC3)n2)=O)CC1 C1(C(=O)NC(C2CN(C(c3ncc(C(C)(C)O)cn3)=O)C2)C)CCS(=O)(=O)C1(C)C CC1=NN(C)C(=O)C1CC(=O)N(C)CC1CCCCN1C(c1cn(C)nc1Cl)=O c1(C(=O)NCC2N(C(COCC(=O)OC)=O)CC2)cc(-c2ccncc2)on1 c1(N2CCC(CC(N3CCC(COC)CC3)=O)C2)nc(OC)cc(C)n1 N1(C(C=C(C)CCc2ccccc2)=O)CCC(NC(C2(S(N)(=O)=O)CC2)=O)CC1C CCC(CC(C)C)C(=O)NCc1nc(CNC(C2CC(SC)C2)=O)cc(O)n1 C#CCCCCCC(C(=O)NC1CCOC1)N(CCS(C)(=O)=O)C c1(C(=O)NC2CCC(NC(CC=CC=C)=O)CC2)cnc2sc(C)cn12 N1(C(c2nc(C)nn2C)=O)CCC(NC(C2CC3CC2C3)=O)CC1C Cc1cc(=NCC(F)CO)[nH]c(=NCCCc2ccc(Cl)cc2Cl)[nH]1 c1(CN2CC(n3ncc(C(=O)O)c3)C2)nc2ccccc2cc1C(F)(F)F C(C)(CO)(C(=O)N1CCCCC1CCCO)NC(C(CO)OC)=O C1(C(=O)NCCC(C=C)C)CC2CC1CC2NC(=O)CCc1cn(C)nn1 C12(C(=O)Nc3cccc(CNC(c4c(C)cccc4)=O)c3)CCC(C1)C2(C)C c1(C(=O)NCC2CCCC(NC(c3cnn(C)n3)=O)C2)cccc2ncnn12 c1(CC(=O)OC)cccc(C)c1C.C1C(Cc2cccs2)S1 c1(C(c2n(CC=C)nnn2)NCc2csc(C(F)F)c2)ccccc1CN(C)C N1(C(C(C)OCCC(C)C)=O)CCC12CN(C(=O)COCCCC(C)C)C2 C1(C)(C(N2CCCC(CC)C2)=O)CCN(C(C2CCOC2(C)C)=O)CC1 C1(CCNC(c2nnc(C(C)(C)C)s2)=O)CCCN(C(C2C3COCC23)=O)C1 C=C(Br)CCC(=O)NC1CC(F)(CNC(C2C3CCCC23)=O)C1 N1(Cc2n(CC)ccn2)CCC2CN(C(c3ccc(Cl)c(CO)c3)=O)CCC12 Cc1ccccc1C(C)C(=O)NC1CCCC1NC(C1CCSCC1)=O c1(CC(=O)NC2CC3(C2)CN(C(c2sccc2Cl)=O)C3)cccc2ncccc12 c1(C(=O)NC2C(C)(C)CN(C(c3cccnc3)=O)CC2)cnn2cccc(F)c12 CCC(CNC(C1(CO)CCN(C(=O)C(C)C2CCC2)C1)=O)CC(C)C N1(C(C)(C)C)CCCC(C)(C(=O)NC2(c3nccs3)CC2)S1(=O)=O C1(NC(=O)CC2(CO)CC2)CCOC12CCN(C(C1CC=CCO1)=O)CC2 Cc1ccc(NC(=O)C(=O)NC2(CN(C)C)CCCC2)cn1 c1(C(N2CCCC(CC=C)(NC(c3csc(C)c3)=O)C2)=O)ccc(N)c(C)c1Cl c1(C(=O)NCC2N(C(CN3CCN(C)CC3)=O)CC=C2)cc2cccn2cn1 C1(CNC(C(C2CCCC2)OCC)=O)CCN(C(=O)CC2CC(CF)C2)C1(C)C C(CC(C)C)(C(=O)N1CCC(CCC(N2CCC(C)(CCO)C2)=O)C1)OC Cc1noc(CC(N2CCC(C(=O)O)CC2)=O)c1C C(C(CC(F)(F)F)NC(c1cn(C(C)(C)C)nn1)=O)NC(CN(C1CCC1)C)=O c1(N(C)CCN2CCCC2)nc(=NCCSC(F)(F)F)[nH]c2c1CCC2 C(CC(C(C)(C)C)NC(=O)C(C)N1CCC1)N(C(c1cc(COC)no1)=O)C C(c1cccc(F)c1)=CC(=O)NCCCOCCN(C(=O)CC1CC(F)C1)C c1(NC(CCC=C(C)C)c2ccccc2)c([N+](=O)[O-])ccc(F)c1I C(CC(C)(C)C)(C(=O)NCC1(O)CN(C(=O)CC2CCCOCC2)C1)OC c1(C(N2CC(N(C(CC(C)C3CCCCO3)=O)C)C2)=O)cc2cccnn2c1 C1(CCOC)CC(NC(C2CCN2C(=O)C(C)=C(C)C)=O)C1 C(=O)(C1=CCC(C)CC1)NC1CCN(C(c2ccc(C#C)cn2)=O)C1CC N1(C(C(C)OC)=O)CC(C2CN(C(c3c(O)cccc3Cl)=O)C2)C1 C#CCC(C)(C)NC(C1(NC(=O)CN(C)C(=O)OCC)CSC1)=O C(=O)(C1=NOC2(CCC2)C1)N1CCC2(NC(c3ccoc3Cl)=O)C(CC1)C2 N1(S(CCCCC)(=O)=O)CCC2(CCCN(C(c3c(F)ccc(C)c3F)=O)C2)C1 N1(C(=O)NCC2C(OC)CC2)CCC(C)(c2cccc(Br)c2)CC1 S(=O)(=O)(c1ccc(Br)c(Cl)c1F)N(CC(c1ccc(Cl)c(Cl)c1)O)C Cc1cc(CNC2CCC(C(=O)Nc3c(C)noc3C)C2)c(C)cc1Br c1(OC)cc(C)ccc1NC(C1CCC1CNC(C1(CC(C)C)COC1)=O)=O c1(OC)ccc(CC(=O)NCC(C)(C)NC(=O)CC(C)(C)C(F)F)cc1[N+](=O)[O-] O=C(CCCCCn1cnnn1)NC12CC1CN(C(c1nc(Br)c[nH]1)=O)C2 n12ncc(F)c1C2.C1(N(CC[Si](C)(C)C)CCO)CCCNCC1 c1(NC(C(=O)NCCCNc2nccs2)=O)ccc(C(F)(F)F)cc1Cl N1(C(C2CN(C(CCOCCOCC)=O)CC2F)=O)CCC(N=[N+]=[N-])CC1 C(=O)(CCC1=NNC(=O)CC1)NCCOCCn1cc(C(CC)OC)nn1 N1(C(c2cc3ccccc3[nH]2)=O)CC2OCCN(C(C3C(F)(F)C34CC4)=O)C2C1 C1(CC(=O)NC2CN(C(CNC(=O)NC)=O)C(CSC)C2)CCC2(CC2)CO1 N1(C(CN(CC)CC)=O)CCCC(n2cc(Cn3ccccc3=O)nn2)CC1 CC1COCCC1N(C)C(C1CCCN1C(=O)C(Cl)Cl)=O O=C(C1=CCCOCC1)N1CCC(c2cccc(CO)c2)C1 N1(C(c2ccc(C)cc2C)=O)CCC2(CC1)COC(CNC(=O)CNC=O)C2 N1(CC(=O)Nc2nnc(O)s2)CCC(CNCc2nccc(C(F)(F)F)n2)CC1 C1(C(C)C)(C(=O)NC(CO)C(F)(F)F)CCN(C(=O)C(F)OC(F)(F)F)C1 N1(CC(C)NC(=O)OCCC(C)C)CCCCC1 C1(CNC(C(F)=CC)=O)COCC2(CCN(C(=O)COc3cccc(O)c3)C2)O1 C1(C(=O)NCCOCCC2CC2)CSCCN1C(C1CN2CCC1C2)=O Nc1cc(C(N2CCC2CNC(=O)C(F)C2CC2)=O)cc(C(F)(F)F)c1 c1(C(N(C2CN(C(Cc3nnc(C)o3)=O)C2)C)=O)c[nH]c(=N)c2[nH]ccc12 C1(C(=O)NCCCN(C(c2cc(C)n(C)c2)=O)C)CCCCC12CC2 c1(CNC2CCCN(C(C3(OC)CC3)=O)C2)cc(N2CCOCC2)ccc1F C(=O)(CCCCCn1cnnn1)N1C(CNC(c2c(C)snc2)=O)COCC1 c1(-n2cc(C(C(=O)NC)N(C)Cc3n[nH]cc3Cl)nn2)ccc(Cl)nc1 C(=O)(C(C)(C)C(=O)NCC1CN(C)CCN1C(=O)CCCCCNC(C)=O)NC C(CNC(c1csc(C(F)(F)F)c1)=O)(C(C)(C)C)NC(C1C(C)CCC1)=O c1(C(C(=O)OC)NC(=O)CCNC(Cl)C(F)(F)F)cc(C)cc(C)c1 c1(C(N2CCC(C(C)NC(=O)C(C)(C)N(C)C)C2)=O)n[nH]c2c1CC1CC21 c1(C(=O)NC(CC)CNC(c2cc(Cl)c(N)cc2F)=O)nccc2cccnc12 Cc1ccoc1C(=O)NCC(C)(C)CN(C(C)C(=O)NCC(F)(F)F)C N1(C(C2CC(CCNC(c3cc(CC)no3)=O)C2)=O)CCCC1(C)COC c1(C(=O)NC(C(CC)C)C(=O)NC)ccn2c(O)nnc2c1 C1(C(=O)NCc2nnc(C)s2)CN(C)CCN1C(=O)C(C)CC1CCCC1 c1(CC)nnc(CN(C)C(C2CC(N(C(=O)CCc3nc(=N)[nH][nH]3)C)C2)=O)o1 C1(CNC(Cc2cnc(OC)nc2)=O)CCN(c2ncncc2Br)CCC1(F)F C(=O)(CCC(=O)OC(C)=O)NC1C(NC(C2(SCC)CC2)=O)CCC1 c1(C(N2CC(NC(c3cccc(N(C)C)c3)=O)C2)=O)cc(N(C)C)cc(C#N)c1 Cc1cc(Cl)cc(N)c1C(=O)NC(C)CN(C(=O)CN(C)C(=O)C1CC1)C N1(C(C=Cc2ccc(C)s2)=O)CC2CCC(CNC(c3n[nH]cc3Cl)=O)(C2)C1 C1(CC(C)NC(=O)CC2CCCNC2=O)CCN(C(c2cncn2C)=O)CC1 N1(C(CCc2nnc(C)s2)=O)CCC2(CCN(c3ncnc4cnccc34)C2)C1 C1(C)(C(=O)NCC2CN(C(c3c(OC)nsc3)=O)C(C)C2)CCCCNC1=O C1(CC)(NC(=O)CCn2cc([N+](=O)[O-])cn2)CCCN(C(=O)CCCC#CC)C1 N1(C(C2(CNC(C3=CCC(C)CC3)=O)CCC2)=O)CC2CCN(C)CC2C1 N1(CC(=O)NC(C(=O)N(c2ccsc2)CC)C)CCC(C)C1 c1(C(N2C(CNC(C3C=C(C)CS3)=O)COCC2)=O)cc(O)cc(F)c1F N1(C(C2(C)CN(C(c3c[nH]ccc3=N)=O)C2)=O)CCC(CF)CC1 C1(CNC(Cc2nccc(OC)n2)=O)NC(=O)CC1(C)C C1(NC(c2n(C)c(S)nc2)=O)CN(C(c2cc(F)c(F)cc2F)=O)CCC1(C)C C1(C(=O)NCC2CC(NC(=O)COCC3CCC3)C2)CC2(C1)CC2F c1(C(=O)NCC2N(C(CN(C3CCSC3)C)=O)CC2)c(O)nnc2c1CCCC2 c1(C(N2C(CNC(c3ccc(C)nn3)=O)C(C)CC2)=O)cnc2cnccc2c1 C1(CC(=O)NCC(CN(C(C=CC(=O)N(C)C)=O)C)O)CC2(CCC2)CO1 C(CCC(C)C)(C(=O)NC(c1ccns1)C)NC(c1cc(C)sc1)=O n1(CCNC(N(C)Cc2ccc(C(C)(F)F)cc2)=O)cc2ccccc2n1 C1(C#N)(C(N2C(CNC(c3n(CCC)ccc3)=O)CCC2)=O)CC1(C)C C1(NC(C(=O)NCC)=O)CCC2CC1CN2C(=O)CN1CCN(C2CC2)C1=O C(=O)(CS(=O)(=O)C1CC1)N1C(C(=O)Nc2ccc(OCC)c(OC)c2)CC(F)C1 c1(C(C)=O)cnc(=NCC2CCCN(C(=O)CNC(c3ccoc3C)=O)C2)[nH]c1 N1(C(COC(CC)(C)C)=O)CCC(C)C1CNC(=O)CN(C)CCO N1(C(COCCCC#C)=O)CC(CNC(=O)C(=Cc2c[nH]cn2)F)CC(C)(C)C1 N1(C(C(CC(C)C)C)=O)CC(CO)C2(C1)CN(C(=O)CC1(C)CCC1)C2 C1(CC#C)(C(=O)NCC2(F)CC(NC(=O)C(F)(F)CO)C2)CCOCC1 C1(CC(=O)NCC(O)CNC(C2(Cl)CC2)=O)CC(C(F)F)C1 C12(C(N3CC(C)(NC(c4cnc(C5OCCO5)s4)=O)C3)=O)CCC(F)(CC1)C2 N1(C(C(c2n(C)c(Cl)cn2)(F)F)=O)CCC2CN(C(C3CC3C(N)=O)=O)CCC12 C(C(C)(C)CC(F)F)NC(=O)NCCC(C(=O)OCC)F C(=O)(C1=CCCCC1C)N(CC(=O)NC1CC1)C1CC1.c12ccc(cc1)[nH]c2=O C(=O)(CC(C)(C)C)N1CC(C(=O)NC(CC(C)NC(C2CC(=C)C2)=O)C)C1 N1(C(C(C)NC(C)=O)=O)CC(CNC(c2ncccc2CO)=O)C(C(F)(F)F)C1 C(=O)(C1=CC2C=CC(C1)C2)N1CC2(CC(NC(C(C)OC3CCOC3)=O)C2)C1 Cc1cnc(F)c(C(N2C3CCC2C(CNC(=O)C=CC2CCOCC2)C3)=O)c1 CCCCC(O)CNC(=O)CSCCNC(=O)CCc1cnc(C)o1 c1(NC(c2cccnc2)CC)cc(NCC2CC2)ncn1 C1(N(C(C(C)OCCOC)=O)C)CCN(C(c2cn(C)nn2)=O)C1 CC1CN(C(=O)C(C(C)(C)C)N(C)C)CCC1C(N1CC(O)CC1CO)=O N1(C(c2cn(C)nc2Cl)=O)CCC(O)C(NC(=O)CN2CC=CC2)C1 C1(C(=O)NC2C(F)CCN(C(c3c(C)cccc3)=O)C2)CCC12CCOCC2 N1(C(C)C)CC(CNC(C2C3CN(C(=O)COc4ccsn4)CC23)=O)CC1=O C1(NC(c2cccc(=O)o2)=O)C2CC1CN(C(c1ccc(C3CC3)s1)=O)C2 c1(C(=O)OC)cccc(CN2CC3(CC3)CC2C(=O)Nc2ccns2)c1C c1(C(=O)NCC(CO)NC(c2c(C)nc(C)[nH]2)=O)cc(Cl)cc(C(F)(F)F)n1 CP(C)(=O)CCC(=O)N1CCCCC1CCNC(C1CCNC1=O)=O N1(C(C2CCCN(C)C2)=O)CC2CCC(C1)N2C(c1nn(C)c(Cl)c1Cl)=O c1(CN(C(C(C)OC2CCCCC2C)=O)C)nc(O)c2ccc(Cl)cc2n1 N1(C(C(C=C)O)=O)CCN(CC2(NC(c3cc(OC(C)C)ccn3)=O)CC2)CC1 c1(CNC2C(C(=O)Nc3ncnc(OC)c3OC)C2)c[nH]c2ncc(Cl)cc12 C1(CC=C)(NC(c2c[nH]nc2C2CC2)=O)CCN(C(C2(CC3CC3)CC2)=O)C1 N1(C(CN(C(=O)OC)C)=O)CCCN(C(=O)C(C)OC2CCCCCC2)C(C)C1 N1(C(c2n(C(C)(C)C)ncc2)=O)CCN(C(=O)OC(C)(C)C)CC12CCC2 C12(C(=O)NC(C3CCN(C(=O)Cc4sccc4Cl)C3)C)CCCC(C)(C1)OC2 c1(C(N2C(C(N3CCC(F)(C(N)=O)C3)=O)CC2)=O)c[nH]c2ccncc12 N1(C(C(CC2CCCC2)NC(Cn2ncc(CC)c2)=O)=O)CCC(N(C)C)CC1 n1(C(C)C)cc(C(=O)NCCn2cc(C(=O)N(C)Cc3cn(C)cn3)nn2)nn1 c1(C(=O)NC2C(OC)C(O)C2)cnc2occc2c1 C(C(O)C(=O)NCCC1(NC(=O)COCc2ccnn2C)CC1)N(C)C N1(C(C2(CC)CC2(F)F)=O)CCC(C)N(C(C2(F)CCCCC2)=O)CC1 C1(C(=O)NC2(CNC(C(C=C)O)=O)CCOCC2)CCC(=O)N(CC)C1 C1(NC(c2c(C)nc[nH]2)=O)CC2(CCN(C(=O)CCc3c[nH]c(=N)[nH]3)C2)C1 N1(C(CC(C)n2ccnc2)=O)CCC2CC1CN(C(C1(CCF)CC1)=O)C2 C1(NC(CONC(CN(C)CC)=O)=O)CC(C)CC(C)C1 C1(C(N2CCCC(C(C)C)(CO)C2)=O)CC2(CCCCCC2)N1 c1(C(=O)NC2CN(C(c3ccc(CC)cc3)=O)C(C)CC2)ncc(C#N)cc1C C1(CNC(CC2C(C)(C)C(O)C2)=O)CCCC2(CN(C(C3CCCCC3)=O)C2)O1 CCCCC(CN=c1cc(C)nc(Cl)[nH]1)NC(=O)C(C)OCC1CCC1 c1(CN2CC(C)(C(=O)Nc3c(C(=O)OC)ncc(Br)c3)C2)cc2ccccc2o1 N1(C(C2CC(OC)(OC)C2)=O)CCC2(C1)CN(C(c1cnc3[nH]ccnc1-3)=O)C2 c1(OC)cccc(C(N2CCCC2C2CCN(C(=O)CN(C)CCO)CC2)=O)n1 c1(N2CCC(CNC(c3c(CC)noc3)=O)CC2)cc(C(F)(F)F)nc(CC)n1 C1(C(C)C)CN(C(=O)Cc2ccccc2)CCC1NC(c1cccnc1N)=O N1(C(C2CC(CC)OCC2)=O)CC2(C1)CN(C(=O)C(C)(C)c1cccnc1)C2 C1(C(N2CC(C3(NC(c4c[nH]ccc4=O)=O)CC3)C2)=O)CCC2(C1)CC2(F)F Cc1ccc(Cl)c(C(N2CCOC(C)(CNC(=O)C(O)C3CC3)C2)=O)c1O O=C1CC2CC(C1)N(C(=O)Cc1ccc(NS(=O)(=O)c3cccs3)cc1)C2 c1(C(N2CC(F)(CNC(C3(CC(C)C)CC3)=O)C2)=O)cn(C)c(=O)nc1O N1(C(c2cc(C)sc2)=O)CC(C2(NC(c3cccc(N(C)C)c3)=O)CC2)C1 C12(C(=O)OC)CCCC(CNC(=O)NC3CNC(C)(C)C3)(C1)OC2 CC1CC(C(=O)NC(CC(=O)NCC2CC(=C3CCC3)C2)C2CC2)CN1C C(C(=O)NCCCON)(C1=CCCCCC1)N1CCN(C(C)=O)C(C)C1 N1(C(Cc2c(C)nsc2)=O)CCCC1C=CC(=O)NCCCOCCO N1(C(c2cc(OC)c(C)cc2)=O)CCN(C(C2CCC(C)O2)=O)CC2(CC2)C1 n1(CC(=O)NC2(CO)CN(C(c3ccnn(C)c3=O)=O)C2)cnc2ccccc12 N1(C(C(CC)CN(C)C)=O)CC(C(N2CCCC2CC(=O)OC)=O)CC12CCC2 c1(C(=O)NC(c2ccc(F)cc2F)CC(=O)OCC)ccc2c(c1N)CCCC2 C1(CNC(n2cnc([N+](=O)[O-])c2)=O)CC2CCC1N(C(=O)CN1CCCC1)C2 CS(C)(=O)=Nc1ccc(C(N2CC3CC3(NC(=O)CCC3CCCCO3)C2)=O)s1 N1(C(C2ON=C(CC)C2)=O)CCCCCC(NC(c2nn(CC)cc2Cl)=O)C1 CC1CCC(c2ccccc2)CN1C(=O)CCC(N)=O.n12cc(nn1)NC(=O)C2 C(=O)(C#CC1CCOC1)NC1C(C)CN(C(C2CC(S(C)(=O)=O)C2)=O)C1 CCC(CC(F)F)C(=O)N(C)CC1CCN(C(=O)C(c2cccnc2F)(C)C)C1 c1(N(C(C2NCC(C(C)=O)C2)=O)Cc2cccc(F)c2)cccc(Cl)c1 N1(C(C(N2C(=O)CCC2=O)CC)=O)CC2CCCC(C1)N2C(=O)CCC1CC1 Cc1cncc(C(N2CC=CC2CNC(=O)Cn2cc(C(F)(F)F)nn2)=O)c1C n1(C(C)C)cnc2c(NC3CCCC3CO)[nH]c(=NC(C)c3ccncc3)nc12 C1(C(=O)NC(C)Cc2cn[nH]c2)CC(N=[N+]=[N-])CN1C(c1n[nH]c2c1CCC2)=O N1(C(c2c(C)nc(N)cn2)=O)CC2CCC(C1)C(NC(c1cccc(O)n1)=O)C2 CC1=C(C(=O)N2CCCC3(NC(c4n[nH]cc4Br)=O)CC3C2)C(=O)OC1(C)C C1(CC(=O)NCC(CN(C(C2CC(O)(CC#C)C2)=O)C)(C)C)CCCCC1C C(CCNC(c1ccnn1C(C)C)=O)(C(=O)NCCCCN=[N+]=[N-])OC O=C(CC(=O)NC1CCCC1NC(=O)C(C1CCCCC1)O)NCC1CC1 C1(NC(Cc2c(CC)con2)=O)CC2CC1N(C(c1ccc(C(F)F)s1)=O)C2 CC(C)C(CN(C)C)C(=O)N1CC(F)CC1C(=O)NCCCC(C)(C)O Cc1ccc2c(c1)C(NC(c1cnc(C)[nH]c1=N)=O)CCC2 c1(C(N2CC3CC3(CNCc3ccccn3)C2)=O)cc(I)ccc1O Cc1nc(Br)sc1C(=O)NCC1C2CN(c3cc(OC(F)F)ncn3)CC12 c1(CNC(=O)NC(c2ccc(Cl)cc2)CC(N)=O)cc2n(n1)CCCO2 CCC(CC)CCCC(=O)NCCCCCN(C(=O)C(C)n1cnnn1)C CC(C)CC(O)C(=O)N(CCC(=O)NCC(c1cccnc1)O)CCCO c1(N(C)Cc2cnc[nH]2)cc(NCCCN2CC3CC3C2)nc(C(F)(F)F)n1 N1(C(C2C(NC(C3(C)CN(C)C(=O)C3)=O)CCO2)=O)CCn2nccc2C1 C1(C(N(CC(C)CNC(C2CC(CC3CC3)C2)=O)C)=O)CCSCC1 c1(CN(C(C=C)C(=O)OC(=O)C(F)(F)F)CCC)nc(C(C)C)n2c1CCCC2 c1(C(=O)NC2C(CNC(C(=O)NC)=O)CCC2)cn(CC(C)C)nc1C(F)F N1(C(c2cc(COC)oc2C)=O)CCC(C)CC1CNC(=O)Cc1ncc(C)s1 C1(C(=O)NCC2(O)CN(C(CC(C)(C)C)=O)C2)CCc2c[nH]nc2C1 CCC(CC(=O)NCCOC(C)(C)C#N)C1CCC1 N1(C(CCC(=O)c2cccnc2)=O)CC(F)(F)CC1CNC(=O)CC1CC12CC2 C1(N2CCN(C)CC2)(C(=O)NC2(C3OCC(C)C3)CC2)CCCCC1 c1(CNC(Cc2cc(C)no2)=O)ncccc1C(=O)NCC1C=CCC1 N1(CC)CCCN(C(=O)CN(C(=O)C(C2CCOC2)OC)CC2CC2)CC1 C#Cc1ccc(C(N2CCC(C)(CNC(c3cnn(C)c3)=O)CC2)=O)c(F)c1Cl c1(COC)ccc(C(=O)NCC2CC(NC(=O)C(C)(CC)OC)C2)cc1 C(C(C)CCCC(C)C)NC(C(C(C)NC(CC=C)=O)C)=O c1(N2CCC(N(C)C(C3CSCC(=O)N3)=O)CC2)nc(=N)[nH]c(Cl)c1[N+](=O)[O-] C1(F)(CNC(=O)Cc2cnsc2)CC2CCC(C1)N2C(C1CCC12CCC2)=O CC(CNC(C1CC1C(F)(F)F)=O)CC(=O)NC(CO)(CO)CO c1(C(N(C(C(N2CCC(CC)C2)=O)C)C2CC2)=O)cnc(C)cn1 CC1CN(c2ncc(F)cn2)CC1NC(=O)CCC1CCCCO1 N1(C(c2nccc(OC)c2F)=O)CC(C)OC2(CCN(CC(N)=O)C2)C1 O=C(CCc1cccc([N+](=O)[O-])c1)N=c1ncn(-c2cccc(F)c2)[nH]1 c1(C(C(=O)NC(CC)CNC(=O)Cn2nnc(=O)[nH]2)O)cn(C)nc1C c1(CC)cc(C(N2CCC2CNC(C2CC=CCO2)=O)=O)cc(O)n1 c1(-c2scc(C)n2)ccc(C(N2CC(C(C)NC(C3COC(=O)O3)=O)C2)=O)cc1 C(=O)(CC(C)P(C)(C)=O)NCCC(C)NC(C1(CC#C)CC1)=O CCCCCCn1nnnc1C(C1(C)CCCO1)NCC(C)(C)C1CCCC1 c1(C(N(CC(C)NC(C2CCC(C#C)CC2)=O)CC)=O)ccnc2ccncc12 CCCCCCCC(=O)NCC(O)CNC(c1ccc(Cl)nc1O)=O C(C(C)(C(=O)N1CC(CNC(=O)CCC(=O)c2ccc[nH]2)C1)OC)OC C1(C(N2CC(NC(C)C)C2)=O)(NC(=O)CN2CCCC2=O)CCCC1C c1(CC(C)C)ccc(C(C)C(=O)NC(C)(C)CCCNC(=O)C(C)C2CC2)cc1 C(=O)(C(C)(C)CS(C)(=O)=O)N1CCN(C(C2CCCC(C)O2)=O)CC(O)C1 c1(C(c2nnnn2CCCOC)NC)ccc(Br)c(Cl)c1.C=CC1(OC)COC1 c1(C(N(CC(CN(C(=O)CCC2OCCO2)C)O)C)=O)cnc(S)[nH]1 CCCCCC(O)CNC(=O)CCC(C)NC(C1(C(=O)OC)CC1)=O C1(C(=O)NC(C2(O)CCN(C(C3CCC4(CC3)CC4)=O)C2)C)CCC2CC2CC1 c1(C(=O)NCC2N(C(CC(C(C)C)C)=O)CC2)cc2cc([N+](=O)[O-])ccc2[nH]1 c1(C(=O)NC(CC)CNC(C2CC(=O)C2C(C)(C)C)=O)conc1C(C)(C)C C1(S(C)(=O)=O)(CN(C2(C)CC(O)(CO)C2)Cc2ccc(OC)cc2)CC(F)(F)C1 C1(C)(C(N(C(CO)C2CC2)C)=O)CN(C(c2cnc(=N)[nH]c2)=O)C(C)(C)C1 N1(C(=O)CCc2ccsc2Br)CCSCC1c1cccs1 C12(CNC(C(C)(C)OCC)=O)CCC(CC1)CN2C(=O)CCc1ncccc1C C1(NC(c2c(COC)nn[nH]2)=O)CCC2(CC1)CCN(C(=O)CCC1CC1C)C2 C1(CC(=O)NC(c2nocc2C(=O)NOCCOCCO)C)COCC1O C1(CNC(c2cncc(C)n2)=O)CN(C(=O)COC(F)(F)F)CCC12CCOC2 N1(C(C2CCN(C(C(COC)O)=O)C2)=O)CC(OC)CC(C)C1 c1(OCC)ccc(NC2CC(COC)C2)c(Cl)c1 C1(C(N2C(CC(=O)N(C)C)CCCC2)=O)CCN(C(=O)C(C)(C)C)CC1O C1(CNC(=O)COCCN(C)C)CN(C(C2CC2c2cccs2)=O)CCO1 C1(NC(C(CN(C)C)O)=O)CC=C(C(=O)NCCC(O)C2CC2)C1 N1(C(CCSCCC)=O)CC(CC(N2CCCCC2C2CC2)=O)C2(CC2)C1 c1(C2C(NC(=NC)NCC(Cc3ccco3)CO)C2)ccc(F)c(C)c1 N1(C(CN(C)C2CC2)=O)CCC(NC(c2coc(Cl)c2)=O)C12CCC2 CC1(C)CCCC(N)(C(=O)NCc2nnc(N3CCCC3)o2)C1 c1(C(N2CC3(C(CNC(C(C)SCC)=O)CC3)C2)=O)cc2c(cn1)COCC2 N1(C(c2cnc(C)o2)=O)CCCCC(C(=O)NCc2ccc(Cl)o2)C1 C1(CNC(C(CC)(C)CC)=O)CCC2(CN(C(=O)C(C)Nc3nc(C)cs3)C2)O1 c1(CN(C2C=C(C)CCC2)C(c2ccn(C)c2-c2nn[nH]n2)=O)ccccc1Cl c1(C(C(C)OC)O)nc(-c2cccc(N(C)C)n2)nn1CCC(C)C C#Cc1ccc(Cl)c(C(N2CCCC2CCNC(C2(CC)COC2)=O)=O)c1 c1(OC)ccnc(C(=O)NCC(c2ccc(F)cc2)NC(C2CCC(=O)N2)=O)c1 C(CO)(CCCCNC(c1cnc(O)c(OC)c1)=O)NC(c1cc(OC)ns1)=O c1(C(=O)NC2CN(C(C(C)(CO)OC)=O)CC2(C)C)cc(C)c(O)c(N)c1 Cc1c(Cl)ccnc1C(N1CCC(Cn2cc(NC(=O)C(O)CC(C)C)nn2)C1)=O C1(C(=O)NCC(O)C(=O)NC2CC(CSC)C2)(CC)CCCCC1 c1(C(C(=O)NCC2CC2)N(CC(C)C)CCC)cc(C#N)n(C)c1 C(=O)(N=c1cc(C)n(C2CC2)[nH]1)C1N(C(c2ccc(C)cc2C)=O)CCC(C)C1 c1(C(=O)NC(C(=O)NC(c2cnc[nH]2)C)c2ccoc2)cccnc1 c1(C(N2CCN(C(Cc3nnc(C)o3)=O)C(C3CC3)C2)=O)ccc(O)c(O)c1Cl N1(C(C2(C)C(C(=O)OC)C2)=O)CCCOC(CNC(C2CC(C)(F)C2)=O)C1 C1(C(N2CC(F)(CNC(c3cc(OC)no3)=O)C2)=O)CCC(C)(C)OC1 n1(CCC(N2CCCCC2Cn2cc(CSC)nn2)=O)c(=O)oc2ccccc12 N1(C(c2ccc(C#N)o2)=O)CCC(C2CCN(C(C3CN(C(N)=O)C3)=O)C2)C1 c1(CC)cccc(C(=O)NCC(C)(O)CNC(=O)CCc2ccc(O)cc2)n1 C1(C)(C(N2CCC(C(N(C)CCOC3CC3)=O)CC2)=O)CCCCC1(F)F c1(C(=O)NC2CCN(Cc3c(OC)cc(F)cc3)CC2F)cc(Cl)c(Cl)cc1O c1(OCC)cccc(C=CC(N2CC(NC(C3OC(C)CC3C)=O)CC2C)=O)c1 C(=O)(CC(C(F)(F)F)NC(c1cccn2cncc12)=O)N1C(C)COCC1 c1(C(C)C(=O)N2CCC2C(=O)NC2CC2c2cnoc2)ccccn1 C12(C(=O)NC(CNC(CC=C)=O)C(C)C(C)C)CCC(C(F)F)(CC1)CC2 c1(C(N2CCCN(c3ncc(Br)c(C(F)(F)F)n3)CC2)=O)ccc(Br)cc1Cl CCCCCCC(O)CCC(=O)OC(C)C(c1ccc2c(c1)CCC(=O)N2)=O NS(=O)(=O)CC(=O)NCC1CCN(C(c2cccc(-c3ccco3)c2)=O)C1 C=CCC(CNC(=O)C=CC(C)C)NC(=O)Cc1csc(Cl)c1 Cc1cccc(CN2CCC(C(N3CC4CCC(C3)O4)=O)C2)c1Br N1(C(C2(C(=O)OC)CC2)=O)CCCC(C(=O)O)CC1.n12cc(nn1)COCCC2 N1(C(C(CC(C)C)OC)=O)CCCN(C(c2ccc3sncc3c2)=O)CC1CO c1(OC)ccc(C(=O)NC2CN(C(c3ccc(Cl)c(Cl)c3)=O)CC2(C)C)c(O)c1 CN=c1[nH]c(C(=O)OCc2nccc(C(F)(F)F)n2)cs1 C1(CNC(=O)C2=CCOC2)(CO)CCN(C(=O)C(c2ccccc2)O)CC1 C1(C(=O)NC2CCN(C(COC(C)=O)=O)C2C)CCCC2(CC2)C1 C1(CC(N2CC(OCCNC(C3CC4(CC4)C3)=O)C2)=O)CCC12CCC2 C1(NC(c2n(C)c(S)nc2)=O)CCC2(CC1)CCN(C(=O)C(F)=C1CCC1)CC2 N1(C(C(=O)NC(C)C)C2CC2Cl)CCC(N2CCOC2=O)C1 C1(NC(C(CCCC)F)=O)CN(C(c2[nH]cnc2C)=O)CC2(CCC2)C1 S(=O)(=O)(CCC(=O)NC1CC2(C1)CC21CC1)NC(C)C c1(NCc2nn(C)c(Cl)c2)nccc(=NCC2CCOCC2(C)C)[nH]1 Cc1nc2ccc(C(=O)NC(CO)CCCNC(=O)C3=CCC(C)CC3)cc2[nH]1 N1(C(CCOCCCNC(CC(C(C)=O)(C)C)=O)=O)CCc2nncn2CC1 C(=O)(C(CCN(C)C)NC(=O)CCOC(C)=O)NCC1(CCC)CCC1 Cc1cc(C)c(C(=O)NC2CC(CNC(c3sc(Cl)c(Cl)c3C)=O)C2)c(C)c1 N1(C(CNS(NC)(=O)=O)=O)CCC(O)(CNC(=O)CC2CCCOCC2)C1 N1(C(c2ccc(F)s2)=O)CC2CCC(C1)N2C(C1OCC2CCCCC12)=O N1(C(C(C2CCCC2)OC)=O)CC(C(=O)NCc2ncccc2O)CC(C)(C)C1 N1(C(C(C(C)C)NC(C)=O)=O)CCN(C(c2ccoc2)=O)CC12CCC2 N1(C(CCS(C)=O)=O)CCC(NC(C2CCCCC23OCCO3)=O)C2(CCC2)C1 CCC(CCC(=O)N(CC)Cc1ccccc1)NC(=O)C=Cc1ccn(C)c1 C(CC(F)(F)C(=O)NNC(=O)C1CC1)n1cc(C2(COC)CCCO2)nn1 C1(CNC(c2cccc(Br)c2)=O)CCCC(NC(c2n[nH]cc2Cl)=O)C1 C(=O)(C#CC(C)(C)C(F)F)N1CCN(CCN(C(C(C)CS(C)(=O)=O)=O)C)CC1 N1(C(c2cnc(C)o2)=O)CC(NC(=O)C=Cc2ncc[nH]2)C(C)(C)C1 N1(C(CCC(C)OC)=O)CCCOC(CNC(c2cc(F)c[nH]2)=O)C1 c1(C(=O)NC2(CNC(C3C(CC)C3)=O)CCOC2)cccn2cc(C)nc12 C=C1CC(C(F)(F)F)(C(=O)NCCCC2CCCN2C(=O)C(F)CC2CCC2)C1 N12CC(CC(F)C1)NC2=O.C1(CN(C(C)(C)C)CC=C)CC(C)C1 N1(C(CCC(=O)NC)=O)CCC(NC(c2cc(C)nn2C2CCC2)=O)C(CO)C1 N1(C(C(C)C)=O)CCC(NC(C2COCCN2CC2CCC2)=O)CC1 N1(C(c2cc(SC)oc2)=O)CCN(CC(=O)NCc2csc(O)n2)CC1 c1(C(N2CCN(C(C3(C#C)CC3)=O)CC2C)=O)cc(F)cc2nccnc12 C1(C(=O)NCCCCCO)CCCN(c2ncc(Cl)cc2Cl)CC1 N1(C(CCOCCOCC)=O)CC(C(=O)NCC(C2(O)CCC2)C)C(C(C)C)C1 c1(OC)ncc(NC(C2C3CC2N(Cc2ccc(Br)nc2F)C3)=O)cc1C#N N1(C(c2nnc(C)s2)=O)CCSCC1CCNC(=O)C(C)Sc1nncn1C N(C1CCc2cc(CNc3nnccc3C#N)ccc21)C(C1C(CC)CCC1)=O C(N=c1[nH]c(=NCC2CCS(=O)(=O)C2)[nH]c2cccnc12)c1cccc(C)c1Br CC(C)C(F)(CNC(=O)Cn1ccnn1)C(=O)NCC1COCCN1C CC#CCC(C(=O)N1CCSC(C)(C)C1)NC(=O)C(C(C)(C)C)OC C12(NC(c3cccc(OC)c3OC)=O)CCCN(C(=O)CC(C)OC)CC1C2 N1(CCNC(CN(CC)CC)=O)CCCN(C(c2cnncc2NC)=O)CC1 C1(C(=O)NCCCOCCCC)C(C)CCN1C(=O)C=Cc1cc[nH]n1 C12(C(=O)NCC(C3CCCC3)NC(C(N3CCOCC3)C)=O)CCCC1C2(F)F c1(C(N(CC(C)NC(C(C2CC(F)(F)C2)OC)=O)C)=O)sccc1C(C)C c1(CC)onc(C)c1C(N1CC(NC(=O)CCCCOC)C(C)C1)=O N1(C(c2c(C)cns2)=O)CCN(C(c2csc(-c3cn[nH]c3)n2)=O)C(C)C1C C1(CNC(C(CCC)C)=O)C2CCC(C2)N1C(c1ccnn1C(C)C)=O CC#CCC(C(=O)N1CCCC(C)(N(C)C)C1)NC(c1cc(OC)ncn1)=O c1(OCC)ccc(C)cc1C(N1CC(n2cc(C(C)(C)OC)nn2)C(C)C1)=O N1(C(COCCCOC)=O)CCC(CO)C(NC(c2cccc(Cl)c2Cl)=O)C1 C(=O)(C(C)(C)C(=O)N1C(C(=O)NCCn2cnnc2C)CC1C)OC c1(C(N(C2CCN(C(CCOC)=O)C2)C)=O)cc(S(N)(=O)=O)ccc1O Cc1c(Cl)sc(Cl)c1C(N1CCC(O)(CNC(c2cnc3n2CCC3)=O)C1)=O CCC(C)(C)CC(=O)N1CCC(CNC(=O)CC2CCOC(C)(C)C2)(OC)C1 Cc1cc(C(=O)NC2C=CC(CC(=O)N(C3CCCCCC3O)C)C2)cnc1O C(CCCCCNC(=O)CCCC#N)N(C(=O)CC1CCC2CC12)C c1(CN2CC(CNC(=O)C3=CCCCO3)OCC2)cncc2ccccc12 C1(C(N(C(C)CNC(c2ccncc2C)=O)CC)=O)CC(=O)c2ccccc2O1 c1(OCCC(=O)NCC(CC)NC(C2(CCN(C)C)CC2)=O)ccccc1Cl c1(C(N2CCOCC2CCO)C(=O)NC(C)(C)C)cc(F)cc2cccnc12 C(=O)(CC(CCC)NC(=O)C(c1cccnc1)O)N1CCN(CCCC)CC1 C1(C(=O)NCC2(F)CCC2)C2CCCC2CN1C(C12COCC1C2)=O c1(SCC)cnccc1C(=O)NCC(CNC(=O)CC1CCC(=O)N1C)OC c1(NC(CC(C)O)=O)cccc(NC(C2(C(F)F)CC2)=O)c1 N1(C(C2C(COC)C2)=O)CC2CCC(NC(c3cnnc(Cl)c3)=O)CC2C1 N1(C(c2[nH]cc(C)c2C)=O)CCC(NC(C2CCCC(CF)C2)=O)C12CC2 Cc1nc(C(N2CC(NC(=O)C(O)CC(F)(F)F)CCC2C)=O)ccc1[N+](=O)[O-] c1(C(N2CC(C)N(C(=O)CC3CNC(=O)O3)CC2)=O)cnc2[nH]ccnc1-2 CC(C(C)(C)NC(=O)CC1CCC1(C)C)NC(=O)COc1ccccc1 c1(OC)cc(C(N2CC3C(C2)N3C(c2nc(Br)cs2)=O)=O)ccc1OC(C)=O n1(Cc2cc(C)on2)nnc(C(=O)NC2(CNC(=O)CN(C)C)CC2)c1C C(=O)(C(C)CC(=O)NC(C1CCN(C(C2(CC(C)C)CC2)=O)C1)(C)C)OC c1(CNC(C(=O)NCCC(=O)NC(C)C)=O)cn(C)nc1O c1(OC)ccc(OC)c(C=CC(=O)NCC2CC(NC(=O)C(C)NC(N)=O)C2)c1 c1(OCC(N2CCCC2c2cn(Cc3cccs3)nn2)=O)ccc(Cl)c(F)c1 N1(C(CCn2ccc(C)n2)=O)CCC(NC(=O)CCc2ccc(C)s2)CC1C C1(CC)COCCN(C(C2(CO)CCN(C(C3CC4CCC4C3)=O)C2)=O)C1 C1(C(=O)NC2C(CNC(c3nc(C)n(C)n3)=O)CC2)C2CCC1(C)C2(C)C N1(C(c2ncn(CC)c2)=O)CC(CNC(=O)C(C)NC(=O)C(C)(C)C)C(C)(C)C1 C1(CNC(C(F)=CC)=O)CN(C(c2ccc(SCCCO)cc2)=O)CC1C CCC(C(=O)NCCC1CCN(C(=O)COCc2nc[nH]n2)C1)c1cccnc1 Cc1ccc(O)c(CNC(=O)NC2CC3CC2CC3c2ccccc2)n1 c1(N2CCC(OCC(C)C)CC2)nc(=NCCc2ccccc2)[nH]c2ccsc12 Cc1ccnc(-c2cccc(C(=O)NCCOCF)c2)n1 C1(CNC(Cc2cc(C)on2)=O)CCCC(NC(=O)CN2CCCCC2)C1 c1(NC(C2CCCC(O)C2)c2n(CC(=C)C)nnn2)cc(C(F)F)cc(CO)c1 C=C=CCCC(=O)NC1CN(C(C2CCCN2c2ccccc2)=O)CC1O c1(CC(=O)NCCC2(CNC(c3sccc3C(F)F)=O)CC2)cccc(Cl)c1F C(=O)(N=c1cc(-c2ccccn2)nc(Cl)[nH]1)N1CCN(C2(C)CC2)CC1 c1(CC)onc(C(=O)N(C)CC2CN(C(=O)C(CC3CCCCC3)OC)C2)c1C C1(CC(N2CC(CNC(C=CCOC)=O)C(C)C2)=O)CCCC2(CC2)C1 Cc1nc(-c2cccs2)sc1C(=O)NC1CCC1CNC(=O)C(C)O C1(CNC(Cc2c(COC)cccc2)=O)CCCC2CN(C(=O)CC3CC3)CC12 Cc1sc(-c2ccccc2CO)nc1C(=O)Nc1ncccc1N(C)C c1(OC)ccc(OC)c(C2CCN(C(=O)C(=O)NCCC(=O)NC3CC3)C2)c1 CC1CN(C(c2ccc(C3CC3)o2)=O)CCC1CNC(=O)CCF c1(OCC)ccc(Cl)c(C(=O)N(CCNC(=O)CSc2cccs2)C2CC2)n1 C1(CN(C(=O)C(CO)NC(=O)C(F)(F)F)C)CCCN(C(=O)C(C)(C)F)C1 c1(CC)ccc(C(=O)N(CC(C)CNC(=O)C(CC)SC)C)c(F)c1 C1(NC(CC(=O)NCC)=O)CCCC(C(=O)N(CC(N)=O)CC(N)=O)CC1 C1(NC(=O)CCC2CCCOC2)CC2CCC1(C(N1CC([N+](=O)[O-])C1)=O)C2 c1(C(=O)NCCC2OCCN(C(C)=O)C2)c(C(F)F)oc(C)c1C CCC(CCOC)C(=O)NCC1CN(C(c2sc(F)cc2C)=O)CC1C c1(C(=O)NCC2(C)CCN(C(c3c(C)cc(C)[nH]3)=O)C2)cnn2c1OCC(C)C2 S(=O)(=O)(c1cccc(NC(C2CCN2)=O)c1)Nc1c(OC)cc(Br)cn1 Cc1ncc(C(=O)NC2CC(C)(NC(=O)CCC3CC3C)C2)n1C c1(-c2cn(COC)nc2)cnc(OCC)cc1C(=O)NC1CC1(F)F C1(CNC(C(C)C#N)=O)CC2CCC1N(C(C1(C)CCCS1(=O)=O)=O)C2 CC(C)CC(C(=O)N1CCC1CN=[N+]=[N-])NC(C1(CC2CC2)CC1)=O O=Cc1sc(CN2CC3(CCN3C(c3cc(F)ccc3I)=O)C2)c(Br)c1Br c1(C(=O)NC2C(NC(c3ncncc3F)=O)CCC2)sc(F)cc1Cl c1(CN2CC(CC#N)N(C(=O)CCCCCl)CC2)cc(F)ccc1[N+](=O)[O-] c1(N(CCS(CC)(=O)=O)C)nccc(=NCC2CC3C(C2)C3(F)F)[nH]1 C(CC(C)C)(C(=O)OC(C)(C)C)NC(CCC)(C)c1nnnn1CC1CCCO1 c1(OC)ccc(NC(=O)CNC(=O)CNC(=O)CC2CC3C=CC2C3)cc1 C1(NC(CCCN(C(=O)OC)C)=O)CC(O)CN(C(=O)C#CC2CCC2)C1 Cc1nn(CC(N2CCC(C(C)NC(C3CCCC3C)=O)CC2)=O)cc1[N+](=O)[O-] C(=O)(C(C)(C)C)N(CC(CNC(C(C)NC(=O)OC(C)(C)C)=O)O)C C1(CN(C(C(F)=C(C)C)=O)C)CCCN(C(=O)COc2ccc(C(N)=O)cc2)C1 C1(CNC(c2sc(Cl)cc2Cl)=O)CC2(CCN(C(=O)C3CC3)CC2)CO1 C1(C(=O)NCCC(=C)CNC(c2cccc(OCC)c2)=O)CCCCC1C CCCC(C(N)=O)NC(C1C=CCN(C(=O)C(C)COC)C1)=O N1(C(C)C)CCC(CC(=O)NCCCOCCN(C)C(=O)NC2CC2)CC1 N1(C(C=Cc2cc(OC)ns2)=O)CCC(O)(CNC(=O)CC2CCC(O)C2)CC1 c1(C(c2ccccc2)CC=C)nc(CCOC(C)C)nn1-c1cccc(C)c1 Cc1nc(=N)[nH]cc1C(=O)NC1CC(C)N(C(=O)CCc2ncc(F)cn2)C1 c1(C(=O)NC(CC=C)CNC(=O)CC2CCCC2)cc(C)c(C)nn1 c1(C(=O)NCCOCCNC(Cc2cncc(C)c2)=O)nn(C)c2c1CSCC2 N1(C(C(C)OCC=C)=O)CC=CC(C(=O)NCC(COC)C(C)C)C1 C12CCCN(C1)C2=O.C1(C#N)(C(=O)NC(C2(n3cncn3)CC2)C)CC1C(F)(F)F c12cc(ccc1Cl)C(=O)NC13CC(C1)(C3)C(=O)N2.c1(SC)ccc(OCC#N)o1 C(=O)(CC(C(F)F)C(C)(C)C)NCC1CCN(C(C(CC(C)C)OC)=O)CC1 O=C1NC(=O)c2c(C(=O)NC3C4CC3N(C(=O)CCN3CCCC3)C4)cccc21 CC1CCCC=C1C(=O)NC(CNC(=O)CN=S(C)(C)=O)CO CC(C)C(C)C(CNC(c1ccccc1Cl)=O)NC(C1CC(Cl)(Cl)C1)=O c1(CNC(=O)Cn2cncn2)ncccc1C(=O)NCC1CN2CCC1C2 c1(CN2CC(C(N3CC(O)C3)=O)(CCO)C2)ccc(OC(c2ccccc2)CC)cc1F C1(CNC(c2c(CC)ncs2)=O)C(C)CCN1C(=O)Cc1ccc(F)cn1 C(=O)(C(C)(C)CC(C)C)N1CCC(F)(CNC(Cn2nc(C)c(Br)c2)=O)C1 c1(-c2cn(CC(=O)NC3C(C(=O)O)C3)nn2)ccc(OCCO)cc1 c1(N(C2CCNCC23CC3)C(Cc2nc(C)sc2)=O)cccc(Cl)c1CO CCC(C)CCC(O)CC(=O)NCC1CC2(CC2)CN1C(c1csc(C)c1N)=O C1(C(=O)NCc2oc(C(=O)NC(CC#CC)CO)c(C)c2)CC2(CCC2=O)C1 c1(C(=O)NCCC2(NC(c3cc(C(C)(C)C)n[nH]3)=O)CC2)ncnc2sccc12 Cc1n[nH]c(C)c1CN1CCNCC1C(=O)NC(c1cccnc1)CCO N1(C(c2coc(CO)c2)=O)CCN(C(=O)C(F)(F)CCn2ccnn2)CC1CO CCCCCCC(C)n1nc(-c2ccc(F)cc2)nc1C1C(C)C1C Cc1ccc(C(=O)NC2CC(C)N(C(C3CCC=CO3)=O)C2)c(O)c1C c1(C(=O)NCCCN(CCCNC(CCC#CC)=O)C)cc2oc(C)cc2[nH]1 c1(C(=O)NC2C(NC(C3(C)CC4CCC3O4)=O)C2)cc([N+](=O)[O-])ccc1O C1(NC(C2CCN(CC(F)F)C2)=O)CCN(C(=O)C2=COCCO2)CCC1(F)F N1(C(CC2CCC(=O)N2)=O)CC(NC(c2nncn2C2CC2)=O)C2CCCCC12 C(=O)(C1CCCn2nccc21)NCC1(C)CCN(c2nnc(C3CCCC3)s2)C1 C(=O)(C1=CCN(C(c2cc(Cl)cn2C)=O)C1)NCC(COC)O c1(CNCCCN(CCCNC(c2ccnc(CO)c2)=O)C)ccc(F)c(F)c1 CC(O)C(F)(F)C(=O)N1CCN(C(c2cccc[n+]2[O-])=O)C(C2CCCC2)C1 C(C(=O)N=c1ccn(CCCO)[nH]1)=CC(C)NC(c1c[n+]([O-])c(C)cn1)=O c1(C(N2CCC2(C)COC)C(=O)NCCOCC)nc(C)co1 N1(C(Cc2cc(OC)c(Cl)cc2)=O)CC2CN(C(C3C(C)C3C)=O)CC2(C)C1 C1(C(=O)NC2C(CNC(=O)Cc3cccc(F)c3)CCC2)CCCCC1(F)F C(C1(C)CCOCC1)=CC(=O)N(CCNC(c1cc(C)c(Cl)s1)=O)CC c1(C(=O)NC2CCCC(N(C(Cc3nc(C)sc3C)=O)C)C2)c(C)nn(C)c1C CC1(C2CCC2)CCCN1C(=O)C(C1CCC1)NC(=O)C(O)Cn1cncn1 C1(CC(=O)NC(CCC=C)C2CC2)CC(C)N(C(c2cccnc2)=O)C1 C1(OC)CCN(C(=O)Nc2nnc(Br)s2)C(C(=O)O)C1 C(CC(Cc1ccccc1)NC1CC1(Cl)Cl)NC(C(=O)NCCn1nnc(=O)[nH]1)=O c1(C(=O)NCC23C(CN(C(=O)Nc4ccc(SC)cc4)C2)C3)cccc(Cl)c1C CC(C)CC(CNC(c1ccc(=O)oc1)=O)NC(c1ccccc1C1CC1)=O CN1CC(C(=O)NC(C(=O)NCCc2cnco2)C2CC2)CC1=O CCC1=C(C(=O)N2CCC2CNC(=O)C(=O)Cc2cccc(Cl)c2)SCCO1 c1(C(C)=O)cc(C(=O)NCC2(O)CC(CNC(=O)CC(C)c3ccco3)C2)co1 C1(NC(CC(CC)OC)=O)CCOC12CCN(C(c1cc(C)cnc1C)=O)CC2 C1(C2CC2)(C=O)CCCCC1.N1(C2CC3CN(C(=O)C(F)(F)F)C2C3)CCCC(F)CC1 C1(C(=O)NCC2C(C(=O)NCc3cc(CC)[nH]n3)CCC2)CCOC(C)(C)C1 c1(C(=O)NC2CCN(C(CC(CCSC)O)=O)C2)cnc2nccnc2c1 S(=O)(=O)(C1(c2cn(CCCC(=O)NC3CCCC3NS(N)(=O)=O)nn2)CC1)NC c1(CCC(N2C(C(=O)NCc3ccc(I)cc3Br)CC2)=O)c[nH]c2ccccc12 C(=O)(C1=CC2CCC1C2)NC1CC2CN(C(c3c(C)n(C)nc3)=O)C1C2 c1(C(=O)NCC2=CCN(C(=O)C=CC(F)(F)F)CC2)cccc2c1CCC2 CC1CN(C(c2cccc(-c3ccccc3F)c2)=O)CC(C)S1(=O)=O Cn1c(O)ncc(C(=O)NCCC2CN(C(C3CSCCS3)=O)C2)c1=O C1(F)(CNC(c2nc(COCC)sc2)=O)CCN(C(C2CCNC2=O)=O)C1 c1(-c2ccc(C(=O)NCc3c(CC)nco3)nn2)ccc(B(O)O)c2nsnc12 c1(C(N2C3C(NC(C4=C(C)CCCC4)=O)C(C3)C2)=O)ccc(C)c2cccnc12 N1(C(C(CCC)OC)=O)CC(C2CN(C(c3c(OC)ccc(Cl)c3F)=O)C2)C1 C1(CNC(CC2ON=C(C)C2)=O)CCCN(C(c2cc[nH]c2C)=O)C1 Cc1c(Br)ccnc1C(N1CCCN(C(=O)CNC(=O)NC2CC2)CC1)=O c1(NC(=O)CC2CN(C(c3cccc(F)c3O)=O)CCO2)ccc([N+](=O)[O-])cc1 C(=O)(CC(C)(O)C(F)(F)F)N.C12CC3(CC13)C(=O)N2.n1(C2CC(OC)C2)cc(C)nn1 C1(C(C)C)(C(=O)NCCCC(O)CO)CCCN1C(C1CC12CCCC2)=O C(=O)(C1=CCOCC1)NC1C(CNC(CCN(CC(F)(F)F)C)=O)C1 Cc1cccc2cc(C(N3CCN(C(=O)C(C)c4cncs4)CC3CO)=O)oc12 C1(C(=O)NCC(CN(C(CCOCC#C)=O)CC)(C)C)CC(C)(C)SC(C)(C)C1 C1(CNC(CN(C(=O)C(C)OCCC=C)CC#C)=O)(COC)CCCC1 C(=O)(C(F)C(=O)NC(C)(CO)C(=O)NCC(=O)N(C)OC)OCC C(CC)(c1ccccc1)=CC(=O)NCC(CNC(C1C(C(=C)C)OCC1)=O)(C)O c1(NC(N2CCCC2CC(c2ccccc2)O)=O)cncc(Br)c1 CC1(C)C=C(C(=O)NCC=CCC(=O)NCC23CCN(CC2)C3)C1 Cc1csc2c(C(N3CCCC(n4cc(CNS(N)(=O)=O)nn4)C3)=O)ncnc12 Cc1cnc(NC2CCCCC2CNC(c2ccc(Cl)cn2)=O)nc1Br CC(C)C(O)C(=O)NC12COC(CNC(C3CCCCS3)=O)(C1)C2 C(=O)(CC(CC)C1CC1)NCC(CC=C)NC(c1cncc(N(C)CC)c1)=O Cc1nccnc1C(=O)NCC1(CN(C)C(C2CC2c2cnc[nH]2)=O)CC1 C1(C(=O)NCC(CC#C)(C)C)C(C2CC2)CCN1C(c1cccc(C)n1)=O C=C(C)C(CC(=O)NC12CCC(C1)N(C(c1cnn(C)c1CC)=O)C2)OCC N1(C(CC2C(C)=NOC2=O)=O)CC2(CCCC2Nc2ncc(I)cn2)C1 C(=O)(C1=CC2(CN(C(c3cc(C)[nH]n3)=O)C2)OC1)NCC(CC)CC(C)C C#C[Si](C)(C)CCCNC(c1cc(Cl)c(Br)s1)=O O(NC(=O)C(C)(F)F)CC(=O)N(C(C)C)Cc1cc(C)on1 Cc1nc(N)c(CC(N2CCOC(CNC(C3COCCN3C)=O)C2)=O)c(O)n1 N1(C(C(CC(C)C)OC)=O)CC2(C1)SCCC2NC(=O)C=CC1CCC1 n1(CC(N2C(CN(C(C3CN(C)C(=O)N3)=O)C)CCC2)=O)ncc2ccccc12 N1(CC(c2ccccc2)CC)Cc2ccc(C(=O)OC)cc2C1 c1(C(=O)NC(CN(C(CNC(CCC)=O)=O)CC)C)occc1C(=O)OC N1(CNCCC2(C)COC(=O)N2)CCC(F)(F)CC1 N1(C(c2cc(CNC(C(CC3CC3)OC)=O)ncc2)=O)CC(=O)NC(C(C)C)C1 C1(C(=O)NCC2(CC)CCCCO2)CCCCN(C(C2(C)CC(C)=NO2)=O)C1 CN1CCn2ncc(C(=O)NCCNC(c3ccc(C4CCCO4)[nH]3)=O)c21 C(=O)(NNc1nc(-c2ccccc2)cs1)c1cncc(C(C)=O)c1 N1(C(C2CCC(C)(C)O2)=O)CCC2(CCCC2NC(=O)C=Cc2cn[nH]c2)CC1 c1(OC)cccc(NC(c2cccc(CNC(C3C4CCC(=O)C34)=O)c2)=O)c1 O(NC(=O)C(O)CCNC(c1cc(C(N)=O)co1)=O)CC(=O)OCC C1(NC(CCN(C)CC)=O)COC2(CCN(C(=O)C(F)n3ccnc3)CC2)C1 CCC(F)(F)C(=O)NC(CCNC(c1cc(-c2ccccc2)ns1)=O)C(C)C N1(C(C(C(C)C)c2cccnc2)=O)CC(C2CCCCN(C(C3(F)CC3)=O)C2)C1 Cc1cc(N2CC(C(C)NC(=O)CCCn3nc(C)cc3C)C2)n2ncnc2n1 Cc1ccc2c(Cl)c(C(=O)NC(C)CCNC(=O)C3=CCCOCC3)sc2c1 CC(C)CCCC(=O)N1CCOC(C(=O)NCCN2C(=O)CCCC2=O)C1 N1(C(CCC2CCC(C)O2)=O)CCC(NC(C2CC(C)(C)C2)=O)C(C)C1 c1(C(=O)Nc2nnn(-c3ccccc3)c2C(F)(F)F)cnn2c1CCC2 c1(C(N2CC(CNC(CCC=C)=O)CC2(C)C)=O)cc(F)c(Cl)cc1Cl c1(C(N2CCC(C)C2CNC(C2CC(F)C2)=O)=O)coc(S(C)(=O)=O)c1 CC(C)C(O)C(=O)NCC1CC(F)CN1C(=O)CC1CC2(CC2)CO1 c1(C(N2C(C)(CNC(C(C)C(F)F)=O)CCC2)=O)ccc2c(c1)CCCO2 C(=O)(CCC(C)OC)NCCCN(C(CC(=O)NC)=O)Cc1ccsc1 C1(NC(c2cc(C)cc(C)c2)=O)CCCC2CN(C(=O)CCC(C)(C)F)CC12 N1(C(CC2(C)CC2F)=O)CC2(CNC(C3(n4nccn4)CC3)=O)CCC1CC2 N1(C(C(CC)OCC)=O)CC(C)(CNC(C23CCCN(CCC2)C3)=O)CC1(C)C C1(C(N(C2CN(C(c3c(CC)cncc3)=O)CC2O)C)=O)CCc2n[nH]cc2C1 C(=O)(C(F)(F)C(F)(F)C(F)F)NCC(CN(C(=O)CCc1nccs1)CC)(C)C N1(C(C(CC)OC)=O)CC2(CC)CC1(CNC(=O)C(c1ccc(C)s1)C)C2 C1(CC(C)NC(C23CCC(C2)C3)=O)CCN(C(C2(C)CCCS2)=O)CC1 O=C(CCCCC(F)(F)F)NCC(C1CCC1)NC(=O)Cc1cccc(F)c1 C1(CC)CCCC1(C)C(=O)NC(C)CC(C)NC(=O)C(C1CCCCC1)O C(c1ccccc1Cl)=CC(=O)NCC(C1CCN(C(c2ncc(Cl)s2)=O)CC1)C N1(C(C2(CC)CC(F)(F)C2)=O)C2CCC(C2)C1CNC(C1CC12CC2)=O Cn1ncc2nc(C(F)(F)F)c(C(=O)NC34CC5CC(C3)C(O)C(C5)C4)cc12 C1(C(=O)OCC)(C(N2CC(NC(=O)C(C)CCN(C)C)C(F)C2)=O)CCOCC1 c1(C(N2CCCC(NC(CC(=C)C)=O)C2C)=O)ccc2nnc(C(F)F)n2c1 C(c1ccc(F)cc1)=CC(=O)NCCCOCCCNC(c1cncc(O)c1)=O c1(NC(c2c(Nc3c(C#N)cnc(C)n3)c[nH]n2)=O)ccc2c(c1)CCCC2=O C1(NC(C(C)C(C)(C)C)=O)CN(C(c2cc[nH]c(=N)c2)=O)CC2(CC2)C1 C=C(C)C1OCCC1C(=O)NCCS(C)(=O)=O N1(C(c2ccnc(OC)n2)C(=O)NC(CC)(C)C)CCC(F)C(O)C1 c1(C(N2C(C)CCC(NC(=O)CCCCCN(C)C)C2)=O)cnc2ncccn12 O=C(C#CC1CCCOC1)NCC1CN(C(=O)CC(F)F)CC1O C1(NC(C(CC)SC)=O)COC2C(NC(c3ccn(C(CC)CC)n3)=O)COC12 C(=O)(N1OC2CCC1CC2)C1C2(CCN(C(C(CC=C)C(C)C)=O)CC2)C1 c1(CC)nc(=N)[nH]c(=NCCC2CCC(NC(c3cccc4nc[nH]c34)=O)C2)[nH]1 N1(C(CCCOCC)=O)CCC2(CC1)COC(CNC(=O)C(C)(C)C)C2 c1(C(N(CCN(C(c2c(CC)ncnc2)=O)C)C(C)C)=O)ccc(C)c(C)c1 C(=O)C#CC1CCCCO1.Cc1cc(C2CCCN2C(=O)C(F)(F)F)ncc1C#N O=C1CC(CC(=O)N2CCN(C(=O)CCc3ccc(F)nc3)C3(CC3)C2)=NN1 Cc1nc2cccnn2c1C(=O)NCC(C)CN(C(=O)CCc1cc(Cl)cs1)C N=c1ccc(C(=O)NCC2CC2NC(c2csc(Br)n2)=O)n[nH]1 C(C(=O)NC(C)CN(C)C(c1cc(C)c(C)o1)=O)(C(C)O)NC(C)=O CC1(C)C(C(=O)NCCCOCCOCCNC(C2CCCC2O)=O)C1(C)C C(=O)(C(C)C(F)F)N(CC(CC)NC(C1(CN(C)CCO)CCCC1)=O)CC CC1=C(C(=O)N2CC3CC3(CNC(C3C(C)(C)C3(C)C)=O)C2)CCC1 C1(NC(=O)CCc2ccccn2)CCN(C(c2cc3occc3s2)=O)CC1O CCN=C(NCC(O)Cc1ccc(Cl)c(Cl)c1)N(C)Cc1ccc(Cl)s1 C1(OC)CCC2(CCN(C(c3cc(CNC(C4CC4F)=O)ccn3)=O)C2)C1 N1(C(C(C)=CC2CC2)=O)CCCC2(C1)C(NC(C1(O)CCC1)=O)CCN2C N1(C(C23C(C)(C)C(CC2)CC3)=O)CCC2CC(C1)CN(C(C1CCOC1)=O)C2 c1(CC(N2CCC(NC(C34CCC3C4)=O)C2)=O)nc(-c2cccnc2)no1 c1([SH](c2n(C3(C)CC3)nnn2)N2CCOCC2)ccc(OC)cc1OCC(F)F N1(C(c2c(C)ncs2)=O)CCCC2(NC(C3CC3c3ccccc3)=O)CCCC12 Cc1cc(CCC(=O)NCCC2(CNC(=O)CC(Cl)Cl)CCCC2)n[nH]1 c1(CC)c(C(=O)NCC(C)(Cn2cccn2)NC(=O)C(C)C(F)F)cccc1F Cc1nocc1-c1cnc(CC(=O)Nc2nn[nH]n2)[nH]1 c1(C(=O)NCC(C(C)C)(C)NC(C2(C3CCC3)CC2)=O)ccc(Cl)c(Cl)c1O C1(C(N2CC3CC3(CNC(=O)Cn3cncc3C)C2)=O)(CC)CCOCC1 N1(C(C(c2ccsn2)NC(=O)OC(C)(C)C)=O)CC(O)(C(N)=O)C1 Cc1ncccc1-n1nc(Cc2ccc(F)cc2)nc1-c1cnc(C(C)(C)C)o1 c1(CCC)nc(C)c(C(N2CC2CNC(=O)CC2CC(c3ccccc3)C2)=O)s1 c1(C(CC)C)ccc(C(=O)NCCC2CCN(C(C3CC4(CSC4)C3)=O)C2)cc1 c1(C(=O)NC2CC(NC(c3ccnc(C)c3C)=O)C2)ccc2sccc2c1 C1(C(C2CC(C(N(C(C3(F)CC3)C)C)=O)C2)=O)CC2C=CCC(C1)C2 C(=O)(CC(C)C(=O)NC1CCCN(C(c2c(C(F)(F)F)nn(C)c2C)=O)C1)OC C1(CC(=O)NC2(CCNC(C(C)(C)NS(C)(=O)=O)=O)CC2)CCC(=O)NC1=O CC(CC1CCCC1)C(=O)NCC1(NC(=O)C(C)OCCN(C)C)CCCC1 c1(OC)ccc(C)c(OC)c1C(N1CCCC(NC(=O)C(O)P(C)(C)=O)C1)=O C1(C(N2CC(CN(C)C(c3cc(Cl)ns3)=O)OCC2)=O)Cc2ccncc2N1 O=C(N=c1cc2ncccn2[nH]1)N1CCC(O)(Cc2ccccc2)C1 C(CO)(C(C)N=c1cc[nH]cc1S(=O)(=O)N1CCCC2(CCOCC2)C1)SC C(=O)(CCCCSC)NC1CC(CC(OC)OC(=O)N(C)C)C1 CCC(CCCO)N=c1[nH]c(=NCC2(OCC)CCSCC2)[nH]c2ncn(C)c12 C(CCCC(CO)NC(c1ccc(C(F)(F)F)o1)=O)NC(c1c(C)n(C)nn1)=O c1(C(=O)NC(C)CN(C)C(c2cncc(C#N)c2)=O)cc2ccc(Cl)cc2[nH]1 C1(CNC(c2c(OCC)scc2)=O)CCN(C(C2CCC(=O)N2CC)=O)CC1 CC(C)(C)C(CO)C(=O)N1CC2(CCC2)CC1C(=O)NCc1csc(O)n1 C1(NC(CC=CC=C)=O)(CNC(C2(F)CCOC2)=O)CCC(C)(C)CC1 c1(C(c2cccnc2)NC(N(CCCN(C)C2CC2)C)=O)ccc2ncsc2c1 C1(CC(=O)NC)C2CN(C(=O)CN(C(=O)CCC3CC3)CCOC)CC12 CC1CN(C(=O)C=C2CCCCC2)CC1NC(c1cscn1)=O CC1=CC(C)C(c2cn(CC(F)CCNC(C3CCC(=O)N3)=O)nn2)CC1 Cc1ccccc1CC(=O)NCC1(F)CCC(NC(c2c(C)ncn2O)=O)C1 n1(CC)cnc2c1CCN(C(C(=O)NCC(F)F)C1CC(OCOC)C1)C2 c1(C(C(=O)NCCCSCC)N(CCF)C2CC2)cc(C)c2ncccc2c1 c1(C(=O)NC(c2ccccc2)CNC(C2CCOC2)=O)snnc1C1CC1 C(C1=CCN(C(=O)COCc2ccc(O)cc2)CC1)NC(C1C=CCCC1)=O C1(CC(=O)N(C2CCCC2(C)O)C)(NC(c2ccncc2Cl)=O)CCCCC1 c1(C(=O)NC(C2N(C(C(CC#C)C)=O)CCC2)C)c(Cl)nc2sc(C)cn12 c1(C(=O)NC23CCCN(C(c4cccc(C)n4)=O)C2C3)cc2sccc2cn1 Cc1cccc2ncnc(NC3CCN(C(=O)Cc4ccon4)C(C)C3)c12 c1(C(=O)NCCC(N2C(CC(C)C)CC2)=O)nnsc1N CCCC(C)C(CC)(c1nnnn1CC)NC1(CO)CCC1 c1(C(=O)NC(CCCC)C(=O)NCc2ccc(O)c(C)c2)cnn2cccc2c1 c1(CNC(C(C)CO)=O)cnn(C)c1C(=O)N(C1CC1)CC1(O)CCC1 N1(C(C(C)OCC#C)=O)CC(C(N2CCCC(O)(C(N)=O)C2)=O)CC(C)(C)C1 N1(c2nc(SC)nc(C(F)F)c2)CCN(C(=O)C(C)C)CC(O)C1 c1(CC(=O)NCCC(C)NC(C(C2CCC2)OCC)=O)ccn(CC(C)C)n1 c1(C(N(C(CNC(CC(COC)(C)C)=O)C)C)=O)cc(OC)c(F)c(F)c1 O=C(C1=C(F)CN(C(C2CN3CCC2C3)=O)CC1)Nc1ccn2nccc2c1 CCC(C)(CC)C(=O)N1CC=CC(NC(c2c(-c3ccccc3)noc2C)=O)C1 C=CC1(CO)CCN(C(C23CCC(CC2NC(=O)CCC(C)C)C3)=O)CC1 c1(C(=O)NCC(C)(CO)NC(CCCC(=O)OCC)=O)cc2cccc(Cl)c2s1 C(=O)(CCCC(=O)NC1CC1)NC(C)CCN(C(=O)CC1CNC(=O)C1)C C1(CCNC(Cn2c(C)nnn2)=O)CCCCN1C(=O)COC1CCOC1 C1(C(N2CCC(N(C(c3cc(CCCOC)on3)=O)C)C2)=O)CC(=O)NC1(C)C C12(CC(=O)NC3CN(C(C4CC(OC)C4)=O)CC3C)CCCN1CCC2 C1(O)(C(=O)NCC2C(NC(C(C)OC3COC3)=O)CCCC2)CCCC(C)CC1 CC1(C(=O)NCC2CCC(NC(c3cccc(C(N)=O)c3)=O)CC2)CCCC1O C1(NC(Cc2cn(C)nc2)=O)CCC(O)CN(C(C2(C3CCCO3)CC2)=O)C1 Cc1cc(C)c2[nH]c(C(=O)NC3CN(C(=O)C(C)(F)C(C)(C)F)CC3C)cc2c1 c1(CN(C(CC)CO)CC(=O)NCc2ccccc2)ccc(C(F)F)cc1 c1(SC)cccc(N2CC(C(=O)NCC3COCOC3)CC2=O)c1 C(C(C)C)(C(O)C(=O)NC1CC(F)CN(C(=O)CCc2ccc(C)o2)C1)OC C1(C)(CC)CCC(C(=O)N(C2CCN(C(c3cc(C)[nH]c3C)=O)CC2)C)O1 Cc1ccc2c(c1)CCC(C(=O)N(CCCn1cc(-c3cccnc3)nn1)C)O2 C(=O)(C1=NOC2COCC12)NC(C1CCCCC1)C(=O)NCC(C)(O)C1CCC1 CS(=O)C=CC(=O)N1CC(OCCNC(c2nsnc2O)=O)C1 C=C(Cl)C(C)(C)C(=O)NCC(c1ccc(OC)cc1)NC(=O)C(=O)NCC C1(NC(c2cc(CO)[nH]n2)=O)CCC2CC1CN2C(c1cc2c(s1)CCOC2)=O C1(CNC(=O)CC2CC(C(F)F)C2)CC2(CCOCC2)CN1C(=O)C1=CCCO1 N1(C(c2ncn(CC)n2)=O)CCCC(O)(CNC(=O)C(=Cc2cccs2)C)CC1 Cc1cc(C(N2CCSCC2C(=O)Nc2cccc(F)c2Br)=O)cc(C#N)c1 c1(CN(C2CC2)CC2CCN(C(=O)OC)C2)ccnc(F)c1Cl C(=O)(CCCCCCn1cc(C(C)O)nn1)NC(C=C)C1CC1 Cc1cccc(C(=O)NCCC2(O)CCN(C(c3ccccc3CO)=O)C2)n1 N1(C(C(COC)C)=O)CCC(C)CC1CNC(c1cnn(C2CC2)c1)=O N1(C(C2C(OC)CCC2)=O)CCCC(NC(c2cccnn2)=O)CC1 c1(C(N2CCC(NC(C3(CC)CCNC3=O)=O)C2C)=O)nc(O)nc(O)c1OC C1(N(C(=O)CC(C)(F)F)C)CCC2CN(C(c3ccncn3)=O)CC12 N1(C(C(=O)NC(C)CN(C(=O)CN2CC3CC3C2)C)C)CCP(C)(=O)CC1 c1(C(=O)NC(CC)CNC(=O)CC2COCC2(C)C)ccc2ncnn2c1 c1(C(=O)NC2CC(NC(C3CCN(CC)C3)=O)C2)cccnc1NS(C)(=O)=O c1(C(=O)NC2CN(C(CCCC(=C)C)=O)C(C)C2)ccc2c(c1)nnn2C CCCCCS(=O)(=O)CC(=O)N1CCCC1CNC(C1C(C(F)F)C1(C)C)=O c1(CC)cc(C(=O)NC(C2CCOC2)CNC(C2CC(OC)C2)=O)ccc1F c1(C(=O)NC2C(NC(=O)CC34CCCC3C4)CC2)cn2cc(Cl)cnc2n1 c1(C(=O)NCC2N(C(C(C)CF)=O)CCOC2)cnc2ccoc2c1 C1(NC(c2cc(N3CCOCC3)cc(F)c2)=O)CC2CCCN(C1)C2 c1(C(N2CC3C(CN(C(C(CCOC)C)=O)C)C3C2)=O)ccc(C(C)=O)nc1O N1(C(C=Cc2cccc(N)c2)=O)CCC2CCN(C(C3(F)CCCCC3)=O)C2C1 n1(CCC)cc(Cl)c(C(N2CCC(N(C(=O)COCCOC)CC)C2)=O)n1 Cc1nc(NC(C)CN(C(=O)CN2CCN(C)CC2)C)c(C)c(O)n1 Cc1nc(Cl)c(NC(=O)CC2CCCN2C(c2ncc(Br)cc2F)=O)cc1Br C1(NC(c2c(CC)noc2C)=O)CC2CC1N(C(c1ccnc(Cl)c1N)=O)C2 C#CCC(CC(F)F)C(=O)N1CCC(CC=C)(C(N2CCC2COC)=O)C1 C1(C)(C(=O)NCC2(NC(c3ccc(C#C)cn3)=O)CC2)CCC(C)(C)CC1 c1(C(=O)NCC2CN(C(c3n(COC)ncc3)=O)C(C)C2)c(C)nc2sccn12 CCC(C(=O)N1CCC(CC(=O)NCCc2nnc(O)o2)C1)C(C)C c1(C(N2CC3OCCN(C(C(C)OC)=O)C3C2)=O)[nH]c2c(c1C)C(=O)CCC2 C(=O)(CC1OCCc2sccc21)N(C1CN(C(C2(O)CC2)=O)C1)C c1(C(N2CCC(C(=O)NC(CN(CC)CC)C)C2)=O)ccc(C)nn1 C1(OC)CC(NC(=O)CCc2cccc(OC)c2)CN(C(=O)CCCCC#N)C1 CCC(C)(C)C(O)C(=O)NC1CCC(NC(=O)C(C)(C)Nc2ccccn2)C1 N1(C(c2cnsn2)=O)CCC(C(N2CCC(CC(F)F)C2)=O)C1 S(=O)(=O)(c1cccc(F)c1)N1CC(C(=O)Nc2cccc(CC)n2)CC(F)(F)C1 C=CCCCC(C1CC1)NC(=O)CC(O)CNC(c1cnn(C)c1C)=O C(=O)(CC(CCN(C)C)CC)NC(CC=C)CNC(=O)CNS(=O)(=O)N(C)C C1(C(c2nnnn2C)NCC2N(C)CCC2)Cc2ccccc2C1 C(=O)(C(F)(F)C(F)(F)F)NC1CC(CNC(=O)CC2CCCC23CC3)C(O)C1 C(C(=O)N1CCC(N(C(=O)CC2CCC(=O)C2)CC2CC2)CC1)(C(C)C)SCC C#CC1CCC(C(=O)NC(CNC(C2COC(Cn3cccn3)C2)=O)CC)CC1 c1(C(=O)NC2CN(C(C(C(C)C)SC)=O)CC2C2CC2)ccc2nn[nH]c2c1O CCCCC(O)C(=O)N1CCCC(N(C(=O)Cc2coc(C)n2)CC2CC2)C1 c1(CNC(C2(C)C=CCCC2)=O)nc(CNC(=O)CC2CCOC2=O)cc(O)n1 Cc1nc(C(=O)NC(C2CCOC2)CNC(c2cnc(C(C)(C)C)o2)=O)c(C)s1 C1(CNC(C2CCN(CC)C2)=O)C2CN(C(=O)CCn3cnccc3=O)CC12 CCCCC(CC(=O)NC1(CO)CCC(C)(C)C1)NC(=O)CN1CC=CC1 CN1C(=O)CCC1C(N1CCOC(CC(=O)NC2CC(n3cncn3)C2)C1)=O C(=O)(C(F)CC(C)(C)C)NCc1c(CNC(C(CC(=C)C)OC)=O)cccc1 c1(CN(CCC)C(C)C)ccc(C(=O)NCCc2[nH]cnc2C)cc1 C1(NC(c2cnc(C)o2)=O)CCCCC1NC(=O)C(F)(F)C1CCOCC1 C1(NC(c2nnn(C(C)(C)C)n2)=O)C2CN(C(=O)CCC(=O)OC(C)(C)C)CC12 N1(C(Cc2c(C)scc2)=O)CC(O)CC1C(N1CC(n2cnnn2)C1)=O N1(C(C(CN(CC)CC)F)=O)CCC(N(C)C(c2n[nH]cc2Br)=O)C2(CC2)C1 C#Cc1ccc(C(=O)NC2CCN(C(c3c(Br)noc3C)=O)C2)cc1Cl C12(C(=O)NCC(CCCC)NC(c3cc(C)[nH]n3)=O)C3C4C1C1C2C3C41C#N CCC(CCC(=O)NC(CO)C(=O)N1CCCC1CC1CC1)OC Fc1cccc2[nH]c(=NCCOCC3CCCO3)nc(N3CCCCC3)c12 Cc1[nH]nc2ncnc(N3CCC3CNC(=O)C(C3CCCCCC3)O)c12 C(=O)(CCC(F)(F)F)NC1(C(N2C3C=CCC2CC3)=O)C(C)CCC1 CCC(O)C(F)(F)C(=O)NCC1(CCNC(c2c(C)noc2C)=O)CC1 c1(CNC(C2CC3CCC2C3)=O)nc(-c2cc[nH]n2)nn1CCOCCO CC1CN(C(c2ncccc2O)=O)CCC1NC(C1CC(n2ccnn2)C1)=O c1(CNC(C(c2cnn(C)c2)NC(CNC(=O)OCC=C)=O)=O)nc(CC)no1 c1(C(=O)NCC2(OC)CCN(C(C34CCCC(C3)OC4)=O)C2)ccc(Cl)cc1F CC#CCCCC(=O)NCC1(NC(=O)Cc2ccc(C)cc2)CCCCC1C C1(CC)(NC(C2(O)CCOC2)=O)CCCN(C(=O)CCN(CCC(C)(C)C)C)C1 c1(CC(N2CC(OC)C(NC(c3cnn(C)n3)=O)C2)=O)ccc(C)cc1Cl N1(C(CCN(C(=O)C(C)CC#N)CC)=O)CCSCC(C)C1 CC1=C(C(=O)N2CCC(NC(c3nccc(F)c3Cl)=O)C2)Cc2ccccc2O1 c1(OCC)c[nH]c(C(=O)N(CCNC(=O)C=C(CC)CC)CCN(C)C)cc1=O c1(C(=O)NC(C)C(CO)NC(=O)CCCC2CCCCC2)cc(S(N)(=O)=O)c[nH]1 CC1CN(C(=O)CC(C)(C)c2ccccc2)CCC1NC(C1CCSC1)=O c1(C(N2C(C)CC(NC(C(C)NC=O)=O)C2)=O)cnc(O)nc1O C(CCCCC(=O)NC(C)(C)C)n1c(-c2ccc(-c3c(C)ncs3)s2)ncc1 c1(C(=O)OC)c(C)cc(C)nc1N1C2CCC1(CNC(C1(CO)COC1)=O)CC2 CC(O)CC(C)(C)CNC(C1(N(C(=O)CCc2ccsc2)C)CC1)=O C1(NC(CCC(=O)OCC)=O)CS(=O)(=O)CC1NC(=O)CCc1ccc(O)nn1 N1(C(c2n(C)ncc2C2CC2)=O)CC2(CCC2NC(c2ccon2)=O)C1 CC1CCN(C(c2csc(-c3cnn(C)c3)n2)=O)C(CNC(C2CCCO2)=O)C1 CC(C)C(C)C(C(=O)NCC=CCNC(c1ncc[nH]1)=O)NC(=O)OC(C)(C)C C1(CCN(C)C)CCN(C(=O)C(Cc2ccoc2)NC(=O)Cn2cccn2)C1 n1(CC2(OC)CCC2)c(N(C)Cc2cccs2)nnc1-c1cccc(C)n1 c1(OC)cccc(F)c1-n1nc(Cc2cccc(F)c2)nc1CC1(C)CC1F CC1(O)CCCC1OC(c1ccc(C(=O)N(c2ccccn2)C2CC2)cc1)=O c1(C(=O)NC(C(N2CCCC(C)(O)C2)=O)CCC2CCC2)cncc2[nH]ccc12 C12(NC(CCC=C=C)=O)CCC(CNC(c3n[nH]c4c3COC4)=O)(CC1)OC2 C(C(CNC(=O)Cc1ccccc1F)C(F)(F)F)NC(c1c(=N)[nH]cnc1)=O Cc1cc(C(N2CCOCC2CNC(c2cc(CN(C)C)c[nH]2)=O)=O)cc(F)c1 C1(C)(NC(CCC2CCN(C(C(C(C)C)C)=O)C2)=O)CC2(CCC2)C1 Cc1[nH]c(C#N)cc1C(N1CC2(CO)CC1(C(=O)NC1(C(F)F)CCC1)C2)=O CC1CN(C(=O)C=Cc2nccs2)CCC1C(=O)NC1CCC2(CC1)N=N2 c1(C(N2C(C)(C(N3CCC(F)(F)CC3)=O)CCC2)=O)cc(Br)c2cc[nH]c2c1 C#Cc1ccc(C(=O)NCC(C)N(C(c2cc(Cl)ccc2O)=O)CC)cc1 c1(OC)cccc2cccc(C(=O)NCCCCNC(C3(F)CCCC3)=O)c12 c1(CC(=O)NC23CCCC2N(Cc2cccnc2)CC3)coc2ccccc12 N(C(=NCCc1ccn(C)n1)NC1CCS(=O)(=O)C1)Cc1n(C)cnc1 O=C(C1=NOC2(CCOC2)C1)N1CCCC1C(c1ccccc1)O c1(C(=O)NCC2CCN2C(c2ccc([N+](=O)[O-])s2)=O)ccn2c1CS(=O)(=O)CC2 N1(C(C(=O)NC)C2CC2(Br)Br)CCN(C(c2cn(C3CCCC3)nn2)=O)CC1 c1(Nc2cccc(CCCC(=O)OC)c2)n[nH]c2ccc(F)cc12 C1(NC(CCc2onc(CC)n2)=O)CC2CC1CN(C(=O)C=CC1CCCO1)C2 C1(C(=O)NC2(C)CCN(C(c3ccc(CO)nc3)=O)C2)C2(CCC2)C12CCC2 C=CCC(CC=C)C(=O)NC1CCN(C(=O)Cn2nccc2N)CC1O C1(C(=O)NCC2C(C(N3C(C(=O)OCC)CCC3)=O)CC2)CCC(C)CC1 C(C)(C)(C(=O)NCCCC1(CNC(=O)Cc2nc[nH]n2)CCCC1)N(C)C c1(C(=O)NCCCN(C(CC2CC(C)(C)C2)=O)CCO)ncn2cc(Cl)ccc12 c1(CNc2ccc(C(=O)Nc3c(NC=O)cccc3)nc2)cccc2c1OCO2 C1(NC(c2cc(SC)oc2)=O)CS(=O)(=O)CC1NC(c1ncoc1C1CC1)=O N1(C(c2cccc(C(C)C)c2)=O)CC(NC(=O)CN=S(C)(C)=O)C2(CCC2)C1 c1(C(=O)NCCC2(NC(C(c3scc(C)n3)C)=O)CC2)noc2c1CCCCC2 c1(C(=O)NC2C(NC(c3n(C)cc(Cl)c3)=O)CCCCC2)ccc(S(C)(=O)=O)o1 c1(CC(=O)OCc2cnn(C3CCOC3)c2)ccc(OC(F)F)c2cccnc12 N1(C(C=Cc2cn(C)nc2)=O)CC2CCC(NC(c3ccccn3)=O)CC2C1 N1(C(=O)CC2CC2C(F)(F)F)CCC2(CCCN2C(c2ccc(=O)n(CCF)n2)=O)C1 C1(C(N2CCC(N(C(CCc3c[nH]c(=N)o3)=O)CCO)CC2)=O)CC(C2CCC2)C1 C(=O)(C(C)C(O)C(C)C)NC(CNC(COC(C)=O)=O)CO N1(C(COCCC)=O)CC(CO)C2(C1)CN(C(=O)Cc1ccc3ncsc3c1)C2 C(=O)(C1=CCCCC1)N1CCCC(Cn2cc(C3CCCN(C)C3)nn2)C1 c1(C(=O)NC2CC(NC(c3nc(C4CC4)ncc3Cl)=O)C2)cccc2nncn12 c1(OC)c(-c2nc(CSc3cccc(OCC(F)(F)F)c3)no2)cccc1C#N c1(NC(c2cn(C(C)C)nc2)=O)cc(F)cc(F)c1.C1C(C)O1 c1(C(=O)NCC2N(C(C3CN(C)C3)=O)CCC2)cc(NS(N)(=O)=O)cc(Cl)c1 C(=O)(CS(=O)(=O)N(C)C)NC1CC(OCC(N2C(C)CCC2)=O)C1 C1(CC(=O)NCC2(CCC)CC2)COCCN1C(C1C=CCCC1)=O N1(C(CC(CC)SC)=O)CCCC(O)(CNC(=O)Cc2ccc(Cl)cc2)CC1 CCCC(C)C(=O)N1CCCC1CN(C(=O)C(C)(C)N1CCOCC1)C C1(NC(CCOCCOC)=O)CC2CC(NC(c3cc(OC)nc(Cl)c3)=O)CC12 c1(C(N(C2CCN(C(C(C=C)O)=O)C2)CC2CC2)=O)ccc(Cl)cc1 c1(C(=O)NC(C)CNC(c2nncn2C2CC2)=O)ncccc1C(F)(F)F CC(CC(=O)c1ccccc1F)C(=O)NC(CNC(C1(F)CC1)=O)CO CC1CCC(C(N2CCCC2CC2CCCO2)=O)N1C(=O)CN1CCSCC1 N1(C(c2cc(C)c(O)cc2)=O)CCn2ncc(CNC(=O)CC3CC34CC4)c2C1 Cc1oc(C)c(C(=O)NC(CC(=O)Nc2ccc(Cl)cc2)C2CC2)c1C N1(C(C2(CCN(C)C)CC2)=O)CCC2(CCC(NC(=O)C#CC3CCOC3)C2)C1 c1(CC(C)NC(CC=C)C2CC2)nnnn1C1CCCCC1 c1(C(N(C)CC2CC(F)(F)C2)=O)c(Cl)cc[nH]c1=N N1(C(C2OCCN(C)C2)=O)CC2CCN(C(c3cnc(C4CC4)nc3O)=O)C2C1 C1(CNC(CC(C)OC)=O)CC2(C1)CN(C(=O)C(C)n1cnnn1)C2 C1(NC(c2cnc(C(F)F)s2)=O)CCCCN(C(c2cn(CC3CC3)nn2)=O)C1 CCC(CCOC)C(=O)N1CC(F)CC1CNC(=O)Cc1cc(OC)no1 O=C1CC2(CCN(C(c3ccccc3F)C(=O)Nc3ccc(Cl)cc3)C2)CN1 N1(C(C2C(NC(COCCC#C)=O)COC2)=O)CC2CCC2C1 C1(C(=O)NC(C2(C(=O)NCc3cscn3)CC2)C)C2COCC12 CCCC(F)C(=O)N1CC(OCCC(=O)NCC2(CCOC)CCC2)C1 C1(CC(=O)NC2CCC(CNC(C(C)=CC3CC3)=O)C2)CCC2(CCC2)O1 N1(Cc2cc(OC)ncc2)CC2(C1)OCc1cc(-c3cccc(C)c3F)ccc12 Cc1ccccc1NC(=O)CC1CC(C)N(C(c2cscn2)=O)C1 CCCC(C)CCN1CCC(COC(C)(C)C)C1 N1(C(c2cc(N)c(F)cc2)=O)C2CCC1CN(C(=O)Cc1cc(F)cc(F)c1)C2 N1(C(C(CCCCC)O)=O)Cc2ccccc2CC1CNC(=O)COCC1CC1 n1(CCC)cc(C(=O)N(C)CCOCCCNC(=O)C(COC)OC)cn1 c1(CC)nc(C)[nH]c1C(N1CCC(CCN(C)C(C2CC2C(C)C)=O)CC1)=O C1(C)(C(=O)NC(C)CC2CCCO2)CN(C(C2CCCCC2)=O)CC1C Cc1nn(C)c(Br)c1C(=O)NC(C1(O)CN(C(C2(CC3CC3)CC2)=O)C1)C c1(C(N2CC(NC(C3CC(C)C3(C)C)=O)(CO)C2)=O)cc(N)cc(F)c1 c1(COC)cc[nH]c1C(=O)NCC1CC(NC(c2ccc(COC)o2)=O)C1 CCC(C(=O)N1CCCC1CC(=O)NCCCc1nc(C)no1)N(CC)CC.O N1(C(C2N(C(C(C)c3ccsc3)=O)CCC2(C)C)=O)CCC12CCC(O)CC2 C#CCN(OC)C(=O)C1(SC)CN(C(c2csc(Cl)c2)=O)C1 N1(C(c2c(OC)cnc(F)c2)=O)CC(NC(=O)C2=C(Cl)CC2)C2CCCC12 N1(C(c2c(C)nsc2)=O)CC(CNC(C2(CF)CC(F)(F)C2)=O)CCC1C [N-]=[N+]=NCC(C(=O)NC1CCCN(O)C1=O)NC(C1CC1(F)Cl)=O N1(C(CC=C)=O)CCC2(CC1)CC2(CO)CNC(c1nn2ccccc2c1Br)=O CCCCCCC(C)C(=O)NC(C)CC1CC2CCC(C1)N2C(=O)C(=O)C1CC1 N1(C(c2c(COC)cco2)=O)CCC(NC(C2(c3ccn(C)n3)CC2)=O)C(C)C1 C(CC(C)(C)C(=O)N(C)CC1(N(C)C)CC1)NC(C(C)n1cncn1)=O C=CCC(C(=O)NCCC1CSCCN1C(=O)C=Cc1cnccn1)NC(C)=O C1(CNCCNC(c2nn[nH]c2C(F)(F)F)=O)C=CCN(Cc2ccccc2)C1 Cc1sc(C(=O)NCC2CCC23CN(C(=O)CCC#N)C3)c(C)c1Br C(=O)(CC(CC)CCCC)NCC(C(=O)N1CC(OCC#C)C1)C(C)(C)C C1(C(C)C)CN(C(N)=O)CCN1CC(c1ccnn1CC1CC1)=O CCCCC(C)C(=O)N1CCC(CN(C(c2nc(C)oc2OC)=O)CC)CC1 N1(C(C(C)c2ccco2)=O)CC(CNC(c2cc(F)c[nH]2)=O)C2(CCOCC2)C1 C1(CC(=O)NC(C2(CNC(c3cc(C4CC4)[nH]n3)=O)CC2)C)CCNC1=O C(=O)(CCCC(=O)Nc1ccccc1C#N)NC(C)C=CC(=O)NCC=C(C)C c1(C(=O)NC2(C)CCC(NC(=O)C3=CCS(=O)(=O)C3)CC2)cccn2nccc12 C1(NC(C2(OCC)CCOC2)=O)CCCC(NC(=O)CC2CC2CC)C1 c1(C(N(C(C)CCNC(=O)CC2(O)CC2)C)=O)cc2c(Br)cccc2s1 c1(OC)ccnc(C(N2CC3CC2C3NC(C2CC2C)=O)=O)c1 C1(CC(=O)NCC(CNC(c2csc(C)c2C2CC2)=O)C)CC2(CCCC2)CO1 C=C(Cl)CC(C(=O)N1CC(c2nocc2C)C1)NC(c1cn(C)nc1CC)=O C1(C)(NC(C(c2ccccc2)OC)=O)CC(NC(C2CC2(C)C)=O)C1 C(=O)(C(C)(O)C(C)C)N1CC2C(CNC(CCCCOC)=O)C2C1 C1(C(=O)NC2C(CC(N3C(CN(C)C)CCC3)=O)CCCC2)C2CCC(F)(F)C12 C1(CC)C(=O)N(C2CCC(c3ccccc3)C2)C(=O)N1C n1(CC(=O)NC2C(NC(COCCCC#C)=O)C2)c(C)cc(C)nc1=O Cc1cc(Cl)c(C(=O)NCc2cn(CCNC(=O)CCC3(C)CC3)nn2)cc1F c1(CC)ccc(NC(=O)CO)cc1.c1(CN(C(C)=O)CC)ncccc1C c1(OC)cc(N)c(C(=O)NC2CCOCC2NC(C2(C)CC3CC3C2)=O)c(F)c1 c1(C(N2CC(COC)(CNC(=O)C(C)(C)c3ccns3)C2)=O)ccc(F)cc1N N1(C(CC2(C=C)CC2)=O)CCN2C(=O)C(NC(c3cnsn3)=O)CC2C1 N1(C(c2c(C)noc2N)=O)CCC2C(NC(c3cnn(CC(C)C)c3)=O)C2CC1 N1(C(C2C=CCCC2)=O)CC2CCN(C(=O)Cc3ccccc3)C2C1 c1(N2C3CC(CNC(CCCC#C)=O)(OC3)C2)nc2ccc(C)nc2s1 CC1(NC(=O)C=C2CC2)CN(C(C2CCCC2O)=O)C1 C(=O)(C1=C(Cl)CCOC1)N1C(C2(NC(c3ccc(C(C)C)o3)=O)CC2)CCC1 c1(C(N(C2CCCN(c3ccncn3)CC2)C)=O)cncc(Cl)c1Cl c1(C(N2CCN(C(c3ccc(C#C)cc3)=O)C(CO)C2)=O)c(C)cc(Br)cc1Cl CN1CCN(C(c2cc(O)ncn2)=O)CC1C(=O)NC1CCN(CC2CC2)C1 C=CCC(C)(C)C(=O)NC(C)CCNC(c1cccc(-c2ccc(Br)cc2)c1)=O N(C(=NCC1(CO)CC12CCC2)NC(C)C)C(C#C)Cc1ccc(Cl)cc1 N#Cc1cc(NC(=O)CC2COCCN2C(c2cnon2)=O)ccc1C(F)(F)F C1(CNC(c2c(C(C)(C)C)ocn2)=O)CCCCN(C(C2CNC(=O)N2)=O)C1 c1(C(=O)NCC(C2CC2)NC(c2ccnc(C)c2C)=O)ccc(N)c([N+](=O)[O-])c1 N1(C(CCCOC)=O)CC(NC(c2ccc(C(N)=O)o2)=O)CC12CCCOC2 c1(C(=O)NC(CCNC(CCc2ccc(C)s2)=O)C)ccc(Cl)c(C(F)(F)F)c1 c1(CC(C)NC(C2OCCOC2C)=O)ccc(CNC(C2CCC2C#N)=O)cc1 C1(C(=O)NCCNC(N)=O)CC(=O)CN1C(=O)C(C1CCCCC1)O Cc1ccc(C(=O)N(C)CC2CN(C(c3c(Cl)n[nH]c3C)=O)C2)c(C2CC2)n1 C1(NC(C(C)C(=O)c2cccc(F)c2)=O)CCCN(C(=O)OC(C)(C)C)C1(C)C c1(CC)ccc(C(=O)NC(C)CCCNC(=O)C(C)N=[N+]=[N-])cc1 N1(C(CC(C)O)=O)C2CCC(C2)C1CNC(c1c(O)cccc1F)=O Cc1ccc(C(N2CC(C)(C)CC2C(N2CCCC(C)CC2)=O)=O)c(C)c1 n12c(N3CCC(Cc4ccc(Br)s4)C3)nnc1C2.C=C(C)CNC.CO CC1CCCCN1CCNC1CCN(CC(=O)O)C1 C1(CNC(C2(OC(C)=O)CC2)=O)CN(C(=O)COC2CCOCC2)C2(CCC2)C1 c1(CC)ccc(F)c(C(N2CC(NC(=O)C(C)OCCC(C)C)C2)=O)c1 Cc1cccnc1CCC(=O)NC1CCCC1CNC(=O)C(N)=O C=C(C)CC(C)C(=O)N(C1CCC(NC(=O)Cn2ccc(C3CC3)n2)CC1)C c1(CCC(=O)NCC2CC(NC(C3(C)CC3(F)Cl)=O)C2)nc2cccnc2[nH]1 N1(c2n(C)nnn2)CC2(CCC(CC(=O)Nc3cnn(CC(F)F)c3)O2)C1 C(C)(CCC(=O)NC(CCSC)C(=O)N(C1CCN(C)CC1)C)OCC c1(C(CN(C)Cc2ccoc2Br)(C)O)ccc(Br)cc1F CCC(CC(F)(F)F)C(=O)N1CCN(C(=O)Cn2cc(C3CC3)cn2)CC(O)C1 C(=O)(C1=CN2CCS(=O)(=O)N=C2C=C1)NC1CC(C)N(C(=O)C=CC2CC2)CC1 C1(F)(CNC(CC2(C=C)CC2)=O)CN(C(C2CN(C(C)=O)C2)=O)C1 CC1C(NC(c2cc(CF)on2)=O)CC2CCC1N2C(=O)C1=CCCS1 CCCCC(C(=O)NC(C1(O)CN(C(c2sccc2C#N)=O)C1)C)N(C)C C1(C(N(C)CCOCCNC(=O)Cn2cc(N)cn2)=O)CCC2(CCCC2)CC1 C1(NC(c2n(CC)ncn2)=O)CCN(C)C(=O)C1.C1COCCOCCOCCO1 C1(NC(C(C)OCCCCCC)=O)(CF)CCN(C(=O)C(C)C(C)C)C1 N1(CC)CCC1C(=O)NCC(C)NC(=O)C(C)N(CC(F)(F)F)C CC(CC(F)F)C(=O)NC(c1ccccc1F)CNC(c1ccc(F)cc1O)=O C1(NC(C(C)NC=O)=O)CN(C(=O)CC2CC(C(C)(C)C)C2)CC12CCC2 C1(C(=O)NCC(COC)(O)CO)N(C(C2CCCC2N(C)C)=O)CCCC1(C)C C(CN=c1[nH]c2c(C)c(C)ccc2s1)NC(c1ccccc1COCCOC)=O c12cc(ncn1)COC(=O)C(C)N2C.c1(NC(c2ccccc2)=O)ccc(Cl)cc1 COn1cnc(C)c1C(=O)NCC1CC1NC(=O)CNC(=O)CC(F)(F)F CN(C)S(=O)(=O)N(C)CC(=O)NC1CC2(C1)CC2NC(C1CC1CF)=O C1(NC(c2cc(OCC)no2)=O)(CNC(c2cc(C)ncn2)=O)CCCCC1C C1(NC(c2cnc(CCC)s2)=O)CCC12CN(C(=O)COc1ccccc1)C2 c1(C(=O)NCC(CNC(COCCCOC)=O)CO)cncnc1C1CC1 C1(C(=O)NCCC(C)NC(C2C3COCC23)=O)CC2(C1)CC2F CC1CCCCC1(CNC(c1cc(C#N)c[nH]1)=O)NC(C1CC12CC(O)C2)=O CCCC(C(=O)NCCN(CC(C)O)C(c1cc(CC)on1)=O)OCC N1(C(c2ccc(CC#C)c(OC)c2)C(=O)NC)CCc2scc(Br)c2C1 N1(C(c2c(OCC)nccc2)=O)CC2(CCC2NC(=O)CC(C)C(F)F)C1 C(=O)(C#CC1CCCCO1)N(C1CN(C(c2cc(OC)c(O)cc2)=O)C1)C CC1(C)OC(=O)C(CC(N2CCN(C(C3(N(C)C)CCCC3)=O)CC2CF)=O)O1 CCC(C)(COC)C(=O)NCc1ccc(C(N2CCC(C)(F)CC2)=O)cn1 c1(C(=O)NCC(C)(C2CC2)NC(C(COC)OC)=O)c(F)ccc(F)c1Cl C1(NC(CCCn2c(C)ncc2)=O)CCCC(NC(c2cncs2)=O)CC1 CC1CC(C(=O)O)CC(C)N1C(c1nnsc1N)=O c1(C(=O)NC(CC(C)NC(c2c(C)ccs2)=O)C)c(Br)nc2n1CCC2 Cc1ccnc(C(=O)NC2CCCN(C(c3ccc(F)cc3)=O)CC2)c1O CCS(=O)(=O)c1ccc(CC(=O)NC2CCCC2NC(c2ccoc2Cl)=O)cc1 C1(N2CCC3(CN(C(=O)CCn4cncn4)C3)C2)CC2CCCCC2NC1=O C1(C(N(CCNC(CC(CC)SC)=O)C2CC2)=O)COC(C)(C)CO1 C(CC(F)F)(C(=O)N1CC(OCC(F)F)C1)N(C(c1ccn(CCC)n1)=O)C c1(C(=O)NC(CNC(C(COC)(C)OC)=O)(C)C)cccc2c1ncn2C C1(NC(C(C)OCCC#C)=O)CC12CCC(NC(c1ccsn1)=O)CC2 C1(CCC)(NC(C)=O)CCCN(C(=O)CCc2nc(C3CC3)no2)C1 N(C1CN(C(C23CCCN(CCC2)C3)=O)CCc2ccccc21)C(=O)CO CCC(C)(C)C(C(=O)N1CC(F)CC1CNC(=O)CCc1ccccc1C)OC N1(C(C(C)OCCCCCC)=O)CC(NC(=O)COCCc2cccs2)C(C)C1 C(CCCCC(=O)N(CC(C)C(=O)NCc1ccc(Cl)o1)C)SC N1(C(C2(C#C)CCCC2)=O)CCC2(CC1)CC(CNC(c1c(C)csc1Cl)=O)C2 N1(C(C2CC(OCC)C2)=O)CC(NC(c2ccc(Br)s2)=O)C(F)C1 c1(-c2cn(CCCOC)nc2)cn2c(n1)CN(C(c1cccc(C#N)c1)=O)CC2 CC(CNC(=O)CC(C1CC1)NC(C1CC=CC(O)C1)=O)S(N)(=O)=O C1(N(C(=O)Cc2c[nH]nc2C)CC)CCCN(C(C2(N(C)C)CC2)=O)C1 Cc1cc(NCc2cnn(CC(F)F)c2)ncc1S(=O)(=O)N1CCC(O)C1 C1(C(NOCC(=O)OC)=O)CN(C(=O)C2=CCCSC2)CC12CCC2 C#CC1CN(C(c2cccc(O)n2)=O)CCN1C(c1cnc(O)c(F)c1)=O N1(C(c2c(C)nn[nH]2)=O)C2CCCC1CC(NC(=O)Cn1nc(O)ccc1=O)C2 C1(CC(N2CCC(OCCNC(c3nc(C)c(C)s3)=O)C2)=O)CCCC2(CC2)C1 N1(C(C2(C(=O)OCC)CCC2)=O)CC2(CCCC2NC(c2cncc(Cl)c2)=O)C1 CC(C)C(CN=C(NCC(F)F)NCC1CC(S(C)(=O)=O)C1)C(=O)OC(C)(C)C CC(O)C(C)C(=O)NCC1CCCC1NC(c1cc(C2CC2)[nH]c1C1CC1)=O C1(C(=O)NCC(CC(=O)NCC(=O)NCC)OC)CCCCC1(C)C C(=O)(C1=CCN(C(=O)CN(C2CCC2)C)C1)N1CC(N(CC=C)C)C1 Cn1cc(C(=O)NCC2CCC2NC(=O)C=Cc2cncs2)c2cccnc12 c1(C(N(CCNC(CCCC)=O)C(C)C)=O)cc(C)n(-c2ccc(Br)cc2)n1 C12(NC(c3scc(C)c3)=O)CCCN(C(=O)CCn3ccnn3)CC1C2 c1(C(=O)NCCNC(c2cnn(C3CC3(F)F)c2)=O)ccc2c(c1)CCCS2 c1(C(=O)NC2(CNC(C(C(C)(C)C)SC)=O)CCC2)cc2c(cn1)NC(=O)CO2 CC(C)C(C)(O)CNC(C1(NC(=O)CC2CCCNC2=O)CCSC1)=O C1(CCCC)CN2CCN1OC(=O)C(C)(F)C2=O.c1(C(=O)OC)cc(C)nc(O)c1 n1(-c2c(C)cccc2)nc(C(=O)NC2CC(C)(NCS(C)(=O)=O)C2)c2c1CCC2 CC1(C)CN(C(=O)C2=CCSC2)CC1CNC(C1(c2cccs2)CC1)=O [N-]=[N+]=NCCCC(=O)NC1CCCC1NC(=O)CCCC1CCCC1 c1(NC(C)=O)ccc(SCCCC(=O)C(C)CF)cc1Cl.N12CCCC1CC2=O CC(CCNC(=O)CNC(C1(C2CCC2)CC1)=O)CCNC(c1ccco1)=O C1(NC(C(C)=CC)=O)CN(C(=O)Cn2cnc(-c3ccccc3)n2)CC1O N1(C(C23OCC(C)(C2)C3)=O)CC(NC(=O)CCc2cnccn2)C(S(C)(=O)=O)C1 C1(C)(CNC(C(CC2CCC2)NC(Cc2ccn(CC)n2)=O)=O)NC(=O)NC1=O C1(C(=O)NC(C2CCOC2)C#C)CN(C(c2cnc(C)nc2)=O)C(C)(C)C1 N1(C(c2cc(SC)oc2)=O)CCN(CCNC(C2CNC(=O)N2)=O)CC1 c1(C(N(C2CCCN(CC)C2)CC#C)=O)cccn2ccnc12 c1(CCC(=O)NC2C(C)(C)CN(C(C3(Br)CC3)=O)C2)c[nH]c2ccccc12 C(=O)(C(CC=C)C(C)C)NC(CCC=C)C(=O)N1CCOC(C)(C)C1 CCC(C)(CNC(=O)C=Cc1cncn1C)C(=O)NC1CC(C)(CO)C1 c1(C(=O)NC2C(CNC(c3c(C)nc[nH]3)=O)C2)c(F)ccc(C(F)(F)F)c1F C1(NC(c2cc(C(F)(F)F)n[nH]2)=O)CN(C(C2CCNC2=O)=O)CC12CC2 N1(C(C(F)=C(C)C)=O)CCCCC(CNC(c2c[nH]cc2C(C)(C)C)=O)C1 CCC(C(=O)NCC(CC(=O)NC(c1cnsc1)C)OC)C(C)(C)CC Cc1cc(C(=O)NC2CCC2CNC(=O)C2CC2)cc(C)c1OC(F)F.O C1(NC(C2ON=C(C(C)C)C2)=O)C(C)(C)CN(C(C2CCCCC2)=O)CC1(C)C c1(C(=O)NC2CC(NC(CN(C(C)C)C)=O)C23CCC3)cc(O)cc(C#N)c1 C=CC(C)(CC)C(=O)NCc1nc(C(N2CC(O)C(O)C2)=O)co1 N1(c2c(C)c(N3CCC(C(N)=O)(N(C)C)C3)ncn2)CCn2c(cnc2C)C1 C1(C(N2CCC(CCNC(CC3(OC)CC3)=O)CC2)=O)CN(S(=O)(=O)N(C)C)C1 c1(C(N2CCC(CN(C(C(C)SC)=O)C)C2)=O)cn(C)cc(Br)c1=O c1(OC)cccc(C(=O)NC2CC(NC(=O)C(C)c3ccsc3)C(O)C2)n1 CCCCN=C(NCc1cc(C)co1)N1CCC(NC(=O)OC)C1 CCCC(CC(=O)N(C)CC1COCCO1)NC(C1CC2(C1)CC(C)C2)=O c1(OC)ccc(NC(C2(C)CCN(C(=O)CCC3(OC)CC3)C2)=O)cn1 n1(CC)nc(C(=O)NCC2COCC2NC(=O)C(=O)NCC(F)F)c2c1CCOC2 c1(CNC2CCN(C(c3cnc(Cl)cc3I)=O)C2)cc(F)c(F)c(F)c1 c1(OCC)ccc(NC(C2(NC(c3c[nH]nc3Cl)=O)CCCC2C)=O)cn1 C1(N(C(=O)COC(C)C)CC)CN(C(=O)Cc2csc(-c3ccoc3)n2)CC1O c1(CC)cc(C(=O)NC23CC2CN(C(c2cn(C4CC4)nn2)=O)C3)ccn1 C1(CCNC(C2CCC(C(N3C(C(N)=O)CCC3)=O)C2)=O)CCCC2CC12 C(CC(C(C)(C)C)NC(=O)C1CC1)N(C(=O)C(c1cc(Cl)ccc1Cl)(F)F)C CC1(C)CC(NC(=O)CC2CCCCCCC2)CN1C(=O)C=C1CC1 c1(C(C(=O)NCCN(C(=O)CCc2cscn2)C(C)C)C)cc2ccccc2o1 C1(C)(COC)CC(NC(c2cc(Cl)cn2C)=O)CN1C(c1csc(C)n1)=O N1(C(C(C)CC2CCCC2)=O)CC(CC(=O)NCC2(CO)CCC2)C2(CC2)C1 N1(C(Cn2c(C)csc2=O)=O)CCC2CN(C(=O)C(c3ccnn3C)C)CCC12 CN1CCC(C(=O)NCc2cnn(C)c2C(=O)NCC(C)(C)N(C)C)CC1=O c1(C(=O)NC(CC)CN(C(=O)CC#N)C)cnn(C)c1-c1ccccc1 CC1(C)CN(C(C2(O)CC2)=O)CCC1C(=O)NCc1ccccc1OC(F)F C(=O)(CS(N)(=O)=O)N1C(CNC(C2CCN(C(=O)NC)C2)=O)CCC1 CC1CCOC(C(N2CCCC(CSC3C=CCC(C(=O)O)C3)C2)=O)C1 C(=O)(NN1CCCC1C(=O)NCC1(O)CC1)C1C(C)(C)C(=O)C1 C=Cc1cnn(C)c1C(=O)NC(C1CCCCN1C(c1cc(Cl)cs1)=O)C C(=O)(C(F)CC1CCCCC1)N(C1CCN(C(=O)Cn2cn[nH]c2=N)C1)C N1(C(CCc2cc(C)[nH]n2)=O)CCC2C(NC(=O)C(C)Cc3ccccn3)CC12 C12(NC(c3c(CC)ocn3)=O)CC(CNC(=O)C(CC)N(C)C)(C1)OC2C C(c1cncc(C)c1)=CC(=O)NC(CC)CN(C)C(c1cc(Br)ccn1)=O c1(C(C)C)ccc(C(C)CC(=O)NCCN(C(=O)CC2CC2(C)C)C(C)C)cc1 C(=O)(C1=COCCC1)NCc1cn(C(COCC)C(=O)NC2CN3CCC2C3)nn1 c1(NC2CN(C(c3c(C(C)C)n(C)nc3)=O)CC2C)cc(O)nc(O)n1 C(CC(=O)Nn1ccccc1=O)C1CCN(C(c2c(C)ccnn2)=O)C1 C1(CO)C(NC(=O)CCC2NC(=O)NC2=O)CCN1C(=O)Cc1ccc(Cl)cc1 Cc1c(C(=O)NCC2(O)CCN(C(=O)CCc3nncs3)C2)ccc2c1CCC2 c1(CC)ncc(Cl)c(C(=O)NCC2(C)CCCN2C(=O)C(O)P(C)(C)=O)n1 c1(C(=O)NC2CN(C(C(CCC)C)=O)CC2O)occ2c1CCCC2 c1(C(N2CC(CC(N3CC=CC3CO)=O)C2)=O)ccc(Cl)c(F)c1 N(C1CCc2cccnc21)C(C1C(C2CN(C(CCS(C)(=O)=O)=O)C2)C1)=O N(C1c2ccccc2OCC1F)CC(=O)NCc1cc(Br)cc2c1OCC2 c1(C(N2CCC(C)(CNC(CC(CC)CC)=O)C2)=O)cc2nc(OC)ccc2[nH]1 c1(N2CCC(N(C(c3ccc4cnnn4c3)=O)CC)C2)cc(S(C)(=O)=O)ncn1 c1(CCC(=O)NCC(C2CCCC2)NC(c2nocc2Cl)=O)nncnc1O CC1(CNC(N2CCOC(c3cn[nH]c3)C2)=O)COC(=O)N1.C(CON)S c1(C(=O)NC(COC)C(=O)NCC2CCC=CCCC2)cccc2[nH]ccc12 C=CC1CC(c2nnnn2CCCC2CC2)(NCC(F)C2CCC2)C1 CN1CCC(C(=O)N2CCC(O)(CNC(=O)C3=CCCS3)CC2)c2ccccc21 c1(C(=O)Nc2cc(C)nn2-c2ccccc2)cccc2c1CC(=O)N2C C1(NC(C(C)(C)OC(C)=O)=O)CCN(C(=O)Cn2cnnc2O)CC1C(N)=O n1(CCOC)cccc(NC(=O)CNC(=O)CNC(c2cnn(C)c2)=O)c1=O S(=O)(=O)(c1ccc(N2CCC(NC)CC2)c(F)c1)NC1C(CC)CCC1.NC N1(C(CN2C(C)CC2)=O)CC(N(C)C(c2ccc(O)c(C(N)=O)c2)=O)C2(CC2)C1 N1(C(=O)NC2CC2c2ccc(Cl)s2)CCn2ncc(-c3ccccc3)c2C1 C1(CC)(NC(c2cnn(CCF)c2)=O)CCN(C(C2CCCN2C)=O)CC1 c1(C(=O)NC2CCN(C(CCC(=O)OCC)=O)C(C)C2)ccc2ccccc2n1 CCC(C)CCC(=O)NC1COCCN(C(C2(n3cccc3)CCCC2)=O)C1 c1(C(N2CC3(CN(C(C(C)O)=O)C3)C2)=O)cccc2nc(O)oc12 CC(CC(=O)NCC(C)(C)CC1CN(C(=O)CCCNC(N)=O)C1)c1cnn(C)c1 CC1CN(C(c2ccc3c(c2)COC3)=O)CC(C)C1NC(=O)C(F)=CC1CC1 C1(CCNC(=O)C(C)Cc2cnco2)(OC)CN(C(=O)Cc2nnc(C)o2)C1 CC1(C)CN(C(=O)CC2(O)CCC2)CC1C(=O)NCC(O)(C1CC1)C1CC1 c1(C(=O)NC(C)CNC(C2(CF)CC2(F)F)=O)ccc2c(c1)nc(O)n2C CCC(C(=O)NCCC(CC)(CC)NC(=O)CN(C1CCSC1)C)C(F)(F)F C1(N(C)C)(C(=O)NC2CC3C(NC(=O)CCCC4CC4)C3C2)CCCCC1 C=C1CCC1(C(=O)NCC1CC(F)(CNC(=O)CC(C)N(C)C)C1)C(=O)OC c1(CC)ccc(F)c(C(=O)NCC2(NC(=O)C=Cc3ccncn3)CC2)c1F Cc1[nH]nc(C(=O)NC(C)CCNC(=O)CCCCc2ccccc2)c1O Cc1occc1C(=O)N(C)CCNC(C1C=CC(NC(=O)OC(C)(C)C)C1)=O c1(C(=O)NC(CNC(Cn2ncc(C#C)c2)=O)CO)c(C)ccc(C)c1C c1(C(=O)NC2C=CCN(C(CCC3C(C)=C3)=O)C2)nc(C)ncc1Cl Cc1cccc(C(N2CCCCC2C(=O)OC(C)C)=O)c1-n1cccc1 C(C(CN=c1[nH]c2c(c(=NCCC(C)c3cn[nH]c3)[nH]1)CCCC2)OC)OC C1(NC(c2cc(Cl)c(Cl)s2)=O)CN(C(c2cnc(Cl)[nH]2)=O)CCC1CO CCC(CC)CCC(=O)N(C(C)CC(=O)N(C1CCN(C)C1=O)C)C N1(C(CCCC(=O)OCC)=O)CCN2CCOCC2(CNC(c2ccoc2)=O)C1 C(=O)(C(C(C)(C)C)N(C)C)N1CC(NC(c2c(C)sc(Cl)n2)=O)(CO)C1 N1(CC(=O)NC(CCC)CNC(c2nsnc2O)=O)CCC(O)CC1 c1(CC(N2C(CNC(COCC)=O)C=CC2)=O)cccc(C#N)c1 CC1C2C(CCN2C(C2CC(=O)NC2(C)C)=O)CN1C(=O)CSCC(F)(F)F c1(C(N2CC(CCNC(C3(COC)CC3(F)F)=O)C2)=O)ccc(C(F)F)c(F)c1 c1(C(=O)NC(C(C)CO)C)cncc(CNC(=O)COCCN(C)C)c1 c1(C(N(CC(O)CNC(=O)CC(C)(C)C2CC2)C)=O)ccc2nn[nH]c2c1 c1(C(=O)NCCNC(=O)CCC2CCCC(O)C2)cc2n(c1)CCCC2 C1(SCC)COCC1N=c1[nH]c(=NCC(=O)NC2CC2)c2ccc(C)cc2[nH]1 C(=O)(CCCCCCC(=O)NCC(C1CC1)NC(=O)CC(F)F)OC C1(NC(c2c(CNC(c3cc(C(C)C)[nH]n3)=O)cnn2C)=O)CCCCCC1O N1(C(CC=CC)=O)CCC(NC(c2ccnc(C)n2)=O)C1C1CC1 c1(CC(=O)NCC(CNC(C(C)CN2CCCCC2)=O)O)c[nH]c2cnccc12 C=CCCC(C)(C)CNC(=O)CCOC1CN(C(C2CC23CCOC3)=O)C1 c1(C(N(CCOCCNC(C(C(CC)O)C)=O)C)=O)cnn2c1CC(C)CC2 c1(C(N2CC(C)C(CNC(c3cncc(C(F)F)c3)=O)C2)=O)c(C#N)cnn1C C12(NC(CN(CCC)C)=O)COC(CNC(=O)CN3CCN(C)CC3)(C1)C2 c1(C(N2CC3=C(CN(C(=O)CC(F)F)C3)C2)=O)cnc2onc(C(C)(C)C)c2c1 n1(C(C)C)ncc2c(NN(C)C3CC3)[nH]c(=NCc3nccc(O)n3)nc12 N1(C(CNC(N)=O)=O)CC2CCCC2(NC(=O)CCCc2ccc(Br)s2)C1 CC(CCN(CCN=[N+]=[N-])C(=O)NC1CSC1)N1CCCC1 C1(CCN(CCCOCc2ccc(OC)cc2)CC)CC(C(=O)O)(CO)CC1O c1(C(C(=O)NC(CC)C)N(C)CC2CCCCO2)sccc1Br C1(NC(C2CCC(C(N)=O)CC2)=O)CN(C(=O)Nc2ccccc2Br)CCC1F N1(C(Cc2cccc(OC)n2)=O)CCC(O)(CNC(=O)Cc2cc(C)[nH]n2)CC1 c1(C(=O)NC(C2CCN(C(c3cccc(F)c3)=O)C2)C)ccc2ncccc2n1 c1(C(=O)NC2CCC(N(C(CC=C)=O)C)C2)ccc(C(F)(F)F)cc1C c1(C(=O)NCC(CC(C)C)NC(=O)CC2CCNC(=O)C2)cc(Cl)ncc1N CCC(C)(O)C(=O)NCC(CCNC(=O)CCCOC(C)C)OC Cc1c(C(=O)NCC(C)(Cn2cccn2)NC(=O)CC2CCCO2)sc(Cl)c1Cl C(N=c1[nH]oc2c1CC(F)(F)CC2)c1c(=O)cc2n(c1)CCC2 N1(C(c2n(CC#C)ccc2)=O)CC2(CCCC2NC(c2cnc(S)nc2)=O)C1 C#CCC(CC#C)C(=O)N1CCC(CO)(NC(=O)Cc2ccc(O)c(C)c2)C1 CCC(CC(=O)NCc1cnn(C)c1C(N1CCOC(C)(C(C)C)C1)=O)C(F)F C=CCCCC(C(=O)NCCOCc1ccc(F)cc1)N1CC2C(C)C2C1 C1(CC=C)(NC(c2cccc(CSC)c2)=O)CCCN(C(=O)C(F)C(C)(C)O)C1 C=CC(C)(C)C(=O)N(CC(C)NC(=O)Cn1ccc(C2CC2)n1)C c1(C(N2CC3(CCCN(C(CCCC)=O)C3)C2)=O)ccc(C)c(S(N)(=O)=O)c1 C1(NC(C(CCC)OC)=O)CCS(=O)(=O)C12CN(C(=O)CSCC)C2 Cc1occ(C(F)(F)F)c1CCNC(N1CCOC(c2cccc(F)c2)C1)=O C1(CC(=O)NCCN(CCC)CC)CN(C(=O)C(C2CCOC2)OC)C(C)(C)C1 C12(C(=O)NCC(CNC(Cc3c(C)non3)=O)C)CCC(O)C1CC2 CC1CN(C(=O)CC#N)CC(C)N(C(c2cccc3c2CCCC3)=O)C1 N1(C(c2[nH]cc(C)c2)=O)CC2COCC(C1)N2C(c1c(C)noc1C(F)(F)F)=O C1(CNC(C2(CO)CCCC2)=O)(CF)CC2(CCC2)C1 N1(C(C2C(C)CCC2)=O)CC(C)CN(C(c2coc(O)n2)=O)CC1C c1(C(CC(=O)N(C2CCN(C(CCCOC(C)=O)=O)C2)C)O)cc(Cl)cc(Cl)c1 c1(C(C(=O)N(CC(CNC(C(C)(CO)OC)=O)(C)C)C)C)cccc([N+](=O)[O-])c1 C1(CC(=O)N(c2cccc(C(F)(F)F)n2)CC=C)CN(C(=O)C2CC2)CCO1 C=C(CNC1CN(C(=O)CC)C1)C1CCOCC1 c1(C(N2CCC(O)(CCNC(CCC(CC)C)=O)C2)=O)cc(N)c(F)c(F)c1F C1(NC(CCc2c(C)noc2C)=O)CCN(C(c2cnsc2)=O)CC1O C1(O)(C(=O)NC2CC(C)(NC(C3CCSCC3)=O)C2)CC2CCC1C2 CS(=O)(CC1CNCCOC1)=NC(=O)CSC1CCC(F)(F)CC1 N1(C(C2C=CCN(C(c3c(C)oc(CO)c3)=O)C2)=O)CCC(C)(C)CC1 C1(C(=O)NCC(C)(C2CC2)NC(=O)CCc2ccc(O)nn2)CCOC(=O)CC1 c1(OC)c(O)cc(C(N2CCCC(F)(CNC(C3(C)CCC3)=O)C2)=O)cc1C#N N1(C(Cn2ccc(C)n2)=O)CCC(NC(c2cc(C(C)(C)C)c[nH]2)=O)C1C1CC1 c1(CC(=O)NC(C)CCCNC(C2(F)CC2)=O)ccccc1[N+](=O)[O-] Cc1cc(C(=O)N(C2CN(C(c3cccc[n+]3[O-])=O)CCC2C)C)cc(F)c1C C1(C(N(CC(COC)C)C)=O)CC(N=[N+]=[N-])CN1C(=O)C(C(C)C)C1CCC1 c1(C(=O)NC2C3CN(C(=O)C(C4CCCCC4)O)CC23)ccnc2ccccc12 C1(C(C)NC(CC2(OC)CC2)=O)CCCN(C(c2cc[nH]c(=N)c2)=O)C1 c1(C(=O)NCC2N(C(CCC(C)OC)=O)CC2)[nH]c2ccc(F)cc2c1C C(=O)(C(C)(C)CC(C)(C)C)N1CC(C(C)C)N(C(C2CN(C)CCO2)=O)CC1 n1(CC(=O)NCC2CCCCN(C(C(CSC)C)=O)C2)ccc2ccc(F)cc12 N#CC1CCC(C(N2CCOCC(C(=O)NCc3nc(CO)n[nH]3)C2)=O)CC1 C1(C(N2CCC(C(=O)NCC(CC)(C)C)(CO)C2)=O)CC(C2CC2)=NO1 c1(C(C)=O)ccc(C(=O)N(C(C)CNC(=O)CC2CCC3CC23)C)o1 C1(NC(c2nc(CC)oc2)=O)CC(F)CN(C(=O)CCCC#N)C1 C1(NC(COC2(C#C)COC2)=O)CCC(NC(C2(C3CC3)CCCO2)=O)CC1 C1(N(C)C)CC2(C1)CC(C(N1CCC(C(N)=O)CC1)=O)C2 Cc1cnccc1OCc1cn(C2CCN(C(=O)C(C)(C)F)CC2)nn1 C1(C(C(=O)NCC(CN(C(CCCOCC=C)=O)C)O)F)CCC(=O)CC1 c1(C(=O)NCCC2(OC)CN(C(=O)CN3CC4CC4C3)C2)cc(Cl)cn1C(F)F C1(C(N2CCC(F)(CNC(C3CNC(=O)N3)=O)C2)=O)CC2CCC1CC2 C1(N(C(=O)CCS(N)(=O)=O)C)CS(=O)(=O)C12CCN(C(=O)Cc1csnn1)CC2 c1(N(CC(C)(C)NC(C2CCCCC2S(C)(=O)=O)=O)CC)ncnc2c1CCCC2 N1(C(C(=O)NC(c2ccccc2)(CC)C)C)C(=O)c2ccc(Br)cc2C1=O CCC(CC(=O)NC1CN(C(=O)CCP(C)(C)=O)CC1CC(C)(C)C)C(C)(C)C C(c1cncs1)=CC(=O)N(C1CCCC1)CCNC(CCOCC)=O N1(C(C(C)OCCCC)=O)CC=CC1CNC(=O)CCCC1CCCCC1 C(CCCCNC(N(C1CC1)CC)=O)OC(=O)NC N1(C(=O)OC(C)(C)C)CC(F)C(F)(C(=O)NCc2ccc(Cl)c(Cl)c2)C1 C1(C(=O)NCCNC(=O)NCC)C=CCCN1C(c1cc(Cl)no1)=O C1(OC)C(NC(=O)CC2CN(C(C3CCCCC3O)=O)CC2C)CC12CCC2 C1(CCC)CCCN(CCCCNC(=O)NC(C)(C)C)C1.C(C)(=O)O C12(C(=O)Nc3ccc(CO)nc3)CCC(CNC(C(CCSC)O)=O)(C1)OC2 CC(C(=O)NCC(C)(C)C)N(CCCN(C)C)C(=O)Cc1cnns1 c1(C(=O)NCC2CCCN(C(c3c(C)noc3N)=O)C2)ccc(F)cc1Cl C1(C(N2CC3CC2C3C(=O)NCCC2COCC2O)=O)(CC)CCCCO1 C1(NC(c2n[nH]cc2C2CCC2)=O)CCCN(C(C2(Br)CC2(F)F)=O)C1 N1(C(C2(CCC)CC2)=O)CCOCC(C(=O)NC(C23CCC(CC2)C3)C)C1 N1(C(C=C(CCC)CCC)=O)CC(C)CCC1CNC(c1cccc(NC)n1)=O c1(NCC(c2ccc(C(F)F)cc2)NC(C2CCC(=O)N2)=O)ccc([N+](=O)[O-])cn1 N1(C(=O)C(N2CC3COC(C2)C3O)=O)CCc2cc(Cl)c(Cl)cc2C1 CC(C)C(C(=O)N1CCN(C(=O)C(C(C)C)n2cncn2)CC1)n1cncn1 c1(NC(C(C(C)NC(C2(O)CCOC2(C)C)=O)C)=O)ccc(O)c(=O)cc1 C12(C(N(C3CN(C(=O)CC4(O)CCCCC4)C3)C)=O)CC1Cc1c[nH]nc12 C#CC1CCCC(CNC(=O)NCc2cc(N)ccc2N2CCOCC2)C1 Cc1n[nH]c(C)c1C(=O)NCC1CCCCC1C(=O)NOCC1CC1 Cc1nc(C)c(CC(=O)NCC2(C)CCN(C(c3c(C)nsc3N)=O)C2)c(O)n1 N12CC3(CCC1CC3)C2=O.Cc1nnnn1CCNC(CO)C(C)c1ccccc1 c1(C(=O)NC2CN(C(c3cc(CC)nnc3C)=O)C3C2C3)ccc(C)c(F)c1F C(=O)(C1CC(C)(C)Oc2ccccc21)N1CC(NC(C(CC)CC)=O)(CO)C1 Cc1cc(C(=O)NCCC(C)NC(c2cc(C3CC3)on2)=O)cc(F)c1C CCC(CC)C(O)CNC(C1CN(C(=O)CC2(C3CC3)CN(C(C)=O)C2)C1)=O C1(C2CCN(C(c3csc(-c4ccco4)n3)=O)C2)(NC(C2CCCO2)=O)CC1 c1(C(=O)NC2CN(CCOC)C(=O)C2)cc(C)c(F)cc1N C1(NC(COCC(=O)NC)=O)CN(C(=O)CC2CC3CC3C2)CC1O CC(CC(F)(F)F)C(=O)NC(C1CCCN1C(c1ccn(CCO)c(=O)c1)=O)C CC(C)C(CN=c1cc[nH]cc1S(=O)(=O)NC(=O)OC(C)(C)C)NCC(C)OC(F)F c1(C(=O)NC2(CCNC(C3C(C)C3C)=O)CCC2)cccc2ccoc12 C1(N(C)C)CC(O)(CNC(=O)C(=O)Nc2ccc(Oc3ccccc3)o2)C1 N1(C(CCOC)=O)CCCCC12CC(NC(=O)C(C)Oc1cccc(N)c1)C2 CCC(C(=O)NC1(C)CC(NC(C2CCCN2c2ccccc2)=O)C1)NC(C)=O C1(C(=O)NC(C=C)C(=O)OC)CCCC(OC)C1.C12(CC1)C(=O)N2 CN1CC2(CN(C(C3C4CC4CN3C(C3CCNC(=O)C3)=O)=O)C2)C1 Cn1nc(-c2cnccn2)cc1NC1CCN(C(=O)C=Cc2ccc(Br)s2)C1 C1(C(N2CCOC3(CC3)C2)=O)CC2CCC(C1)N2C(C1(Cl)CCC1)=O CC1CC(NC(c2cnc(O)o2)=O)CN(C(c2scnc2C(F)F)=O)C1 C1(NC(C(C)N(C(CC2C(CC)C2)=O)C)=O)CC2(CCCO2)C1 Cc1cc(Cl)c(C(N2CCCC2C(C)NC(c2cnn(C)c2C(C)(F)F)=O)=O)s1 c1(C(=O)NCC(CNC(c2ccn(C3CC3)n2)=O)OC)cccc(C(C)(C)C)n1 c1(CC)c(C(=O)NCC(C)(C2CC2)NC(=O)C(C)CCOC)cnc2ncnn12 CC(C)(CCNC(C1(CCF)CC1)=O)NC(c1ccc(-c2cccs2)o1)=O C(=O)(C(C)C(=O)NC1CC(CC(=O)NCC#CCCO)C1(C)C)OC CC1CC(NC(c2cnn(C)c2)=O)CN(C(C2CCCCC2(C)C)=O)C1 N1(C(c2nnc3ccccc3n2)=O)CCOC2CN(C(C34COCC3C4)=O)CC12 C(CCCC(C)(C)NC(=O)Cc1ccco1)NC(COCC)=O Cc1ccc(CC(=O)N(C(C)(C(=O)NC(C)CCn2cncn2)C2CC2)C)cn1 c1(NC(CC=C)C)cc(S(=O)(=O)NCc2nc(C)sc2C)ccc1C#N CCCCC(C(=O)N(C)CCNC(=O)CC1CCC(C)(C)CC1)NC(N)=O C1(C(=O)NC2(C)CN(C(CCC)=O)C2)CC2CCCC(C1)C2=O c1(OCC(=O)NCCC2N(C(CCC=C)=O)CCOC2)cc(Cl)ccc1Cl C1(C(=O)OC)CN(C(=O)CCCc2ccc(O)cc2)CC1C(=O)OC c1(C(=O)NC(CC)CN(C(=O)Cc2cscn2)C)ccnc(N2CCCC2)n1 S(=O)(=O)(c1cnc(NCCc2cnoc2)c(Cl)c1)N1CCCCC(SC)C1 N1(C(c2c(CC)nccn2)=O)CC(CNC(=O)C(C)(C)CNC(C)=O)CC1(C)C c1(CNC2C3CN(C(=O)CCCCO)CC32)ccc2ccsc2c1 c1(CC)cnc(C(=O)NCc2ccc(C(=O)NCC(C)(CO)N(C)C)o2)nc1 CC1CN(C(c2ccccc2F)=O)CC1CCNC(C1CC12CCCC2)=O CN(CC1CCC2(CCC2)O1)N1CCCC(F)(c2ccccc2)C1 C(CC(C)(C)C(=O)NCC1C(CO)C1(F)F)NC(c1c(C)coc1)=O C1(c2nnnn2C2COC2)(NC2(S(CC)(=O)=O)CC2)CCCN2CCSCC12 c1(-c2cn(CC(=O)N(CCC3CC3)CC3CC3)nn2)cccc(OC(F)(F)F)c1 CC1OC2(C(=O)NCC3CCN3C(=O)CC=CC(C)(C)C)CCC1CC2 c1(OC)ccc(C(C)NC2(C)CCSCC2)cc1Br c1(C(N(C2CCN(C(c3c(NC)cncc3)=O)C2)C)=O)cc2nc(C)sc2[nH]1 c1(CC)ccc(C(N2CC(CNC(c3cc(C(N)=O)c[nH]3)=O)C(C)C2)=O)cn1 N1(CC)CCCCC1C(=O)NCC(F)CNC(C1C2(CC2)C12CC2)=O c1(C(N2CCC(N(C(=O)C(C)C3CC3)CC#C)CC2)=O)ccc(C(C)C)c(O)c1 C1(NC(CCc2cnc(C)s2)=O)CN(C(=O)CCSCC(N)=O)C2(CCOC2)C1 c1(NC(=O)C#CCNC(c2ccc(O)c(F)c2)=O)cnc2[nH]cnc2c1 Cc1[nH]nc2ncc(C(=O)NCC(C)CNC(C3CCC(=O)N3C3CC3)=O)cc12 C1(C(N2CCC(CN=[N+]=[N-])C2)=O)(NC(C2C(C(C)C)CCO2)=O)CCCCC1 C1(CNC(C(CO)NC(N)=O)=O)CC2CN(C(C34CC(CC(F)F)(C3)C4)=O)CC12 C1(C)(NC(C(=O)N(C)C)=O)CCN(C(=O)C2CC2)C1 c1(C(N2CC(C)(NC(C(N3CCOCC3)C)=O)C2)=O)c[nH]c(=O)cn1 Cc1[nH]c2ccc(C(=O)NCC3CCCCN3C(c3sccc3F)=O)cc2c1C C1(C)(C(N(CCNC(c2coc(COC)n2)=O)CC)=O)CCC(=O)N1 c1(C(N2C(CCNC(C(C)(C3CC3)OC)=O)CCC2)=O)ccc(F)c2[nH]ccc12 N1(C(CN2CCC(C)C2)=O)CCC(C)N(C(c2cc(-c3ccco3)cs2)=O)CC1 C1(=CC(C(=O)NCC2N(C(CCSC)=O)CC2)=O)CCCCC1 C1(OC)CCCC(NC(c2nscc2C(=O)Oc2cnc(C)cn2)=O)C1 c12ccc(o1)C(=O)NC2.c1(C2CN(C(C=CC(C)(C)SC)=O)C2)[nH]nnc1C c1(CSCc2c(OCC)cc(Cl)cc2)c(C)cc(C)cc1C C(=O)(C(C)CCOCC)NCC1(CNC(C2(OC)CCOC2)=O)CC1 N(C(=NCCSc1ccccc1)N1CCC2(CC(C(F)F)=NO2)C1)CC(C)(C)C C1(NC(C2CC(C#N)(OC)C2)=O)CCCN(C(c2ncccc2SC)=O)C1C C#CCC(CC(F)F)NC(C1CCOC1CNC(C1(C)CCC1)=O)=O c1(C(=O)NC2(C3CCCN3C(=O)C(O)C(F)F)CC2)nnc(O)nc1O C1(Cl)(C(N2CC(c3cn(C(C)CSc4ccccc4)nn3)C2)=O)CC12CCC2 N1(C(C(C)(C)c2cccs2)=O)CC2CCCC2(NC(=O)CC2CCCOC2)C1 c1(C(C(=O)NC(CN(C(C(C)NC(CC)=O)=O)C)C)(C)C)cc(Cl)ccc1F C1(C2CCN(c3nc(C)ccc3C(=O)OC)CC2)(NC(C=COCC)=O)CC1 C1(NC(c2cc3ccc(Br)nc3[nH]2)=O)CCCC2(CCCCC2)C1 CCC(CC(C)C)C(=O)NCC1CCN1C(=O)Cn1cc(C)ccc1=O c1(CC(=O)NCC2CC(NC(C3C(CC)CCC3)=O)C2)ncn2c1COCC2 CC(CCc1ccccc1F)C(=O)NCC1CCN(C(=O)CC(F)(F)F)C1 CC1(NC(C2(C(=O)N(C)C)CCC2)=O)CN(C(C2CCC(OC(F)(F)F)C2)=O)C1 Nc1c(F)ccc(Cl)c1C(=O)NCCC1(NC(=O)CCCC2CC2)CCCC1 N1(C(C2(N(C)C)CC2)=O)CCC(F)(F)C(CNC(C2(C3CC3)CC=CC2)=O)C1 C1(NC(=O)C(C2CCCCC2)F)CC2CCC(C1F)N2C(c1ccc(O)cc1)=O N1(C(C(N)COCc2ccccc2)=O)CCNC2(CCNCC2)C1 c1(C(N2C(CN(C(CCCOCC)=O)CC)CCC2)=O)ccc(Cl)c(C)c1N C12(NC(c3nn(C)c(Cl)c3Cl)=O)CCN(C(C3CCCCC3)=O)CCC1C2 C(C(=O)NC1(C)CC(NC(C2CC2c2cccc(Cl)c2)=O)C1)(C(C)C)OCC C=CCC(CNC(=O)C(C)(C)CC=C)C(=O)Nc1ccccc1C N1(C(c2cccc(SC)c2)=O)CC2CN(C(=O)CCc3cc(C)[nH]n3)CC12 N1(C(=O)CCC2CCC2)CCC(C(N2CCC(O)(CO)C2)=O)(CF)C1 c1(C(C)(C)C)ccccc1NC(C1CC1NC(c1ccc(F)nc1)=O)=O N1(C(C2(CC)CCOC2)=O)CC2(COC)CC1(CNC(=O)CCC(N)=O)C2 C1(NC(C2(OC)CCSC2)=O)CCCCC1C(=O)NC(c1cn[nH]c1)C C1(C(=O)NC(C2CCCC2)CNC(C(CC)C(C)C)=O)CN(S(=O)(=O)N(C)C)C1 CCN=c1[nH]cc(C(N2CCCC(NC(C3CC3c3cccc(C)c3)=O)C2)=O)s1 c1(C(N2CC(NC(CN(C3CCSC3)C)=O)C(F)C2)=O)cc2c(F)cccc2[nH]1 CC1CN(C(=O)C(CCN(C)C)c2ccccc2)CCC1CNC(=O)C1=NOCC1 C1(C)(CC)CC(NC(c2cc(C(N)=O)co2)=O)CN1C(=O)CC1CCSCC1 C1(C(N)=O)CN(N2CCOc3c(Cl)cccc3C2)CC1c1ccccc1 C1(C(=O)NC(COCC)C)CC2(CCN(C(C34CCC(C3)OC4C)=O)C2)C1 C1(C(=O)NC(C2CC(=O)NC2=O)(C)C)CCN(C(=O)Oc2ccccc2)C1(C)C c1(CC(=O)NCC2(C(=O)NCCC3(O)CCCCC3)CC2)ccc(O)nc1 C1(C(N(CC(N2CC(C=C)C2)=O)C)=O)(NC(=O)NC)CCOCC1 N1(C(C2N(C(C)=O)CSC2)=O)CCN(C(=O)CN2C(C)CCC2C)CC(O)C1 c1(OCC)nc(N(C2CN(C(c3coc(Cl)n3)=O)C2)C)ncc1C N(C1c2ccccc2CC1NC(=O)CSC(F)(F)F)C(C1C(C=C)C1)=O C(C)(CN=c1nc(C)c(C)c(C)[nH]1)(C(C)C)OC N1(C(C(CN(C)C)(C)C)=O)CC(C2CN(C(C3CCC3c3nc[nH]n3)=O)C2)C1 CCC(C)C(C(=O)NCC1(C)CCCCC1O)NC(=O)CN1CC2CCC1C2 C1(C(=O)NC2CC(CNC(C3CCCNS3(=O)=O)=O)C2)CCc2cncn2C1 N1(C(Cn2c(C)cc(C(F)F)n2)=O)CCC(C2(NC(=O)CC(C)C(F)F)CC2)C1 N1(C(C(C)NCc2ccco2)=O)CCCCC1CN c1(OC)ccc2c(c1)CC(C)CC2NC(=O)NCCOc1cccc(O)c1 N1(C(c2cncs2)=O)CCCC(C2CCCCN2C(c2ccc(Cl)nc2)=O)C1 C(=O)(C(O)P(C)(C)=O)NC1C(N2CCN(C(CSCCC)=O)CC2)CCC1 C1(CC=C)(NC(=O)COCC(C)C)CCN(C(=O)CC23CCCC2C3)CC1 C12(CNC(Cc3n(C)ccn3)=O)CCCCC1N(C(C1CC13CCC3)=O)CCC2 c1(C(=O)NC2C(NC(CSCc3nnc(C)s3)=O)C2)ccc2c(c1)CN(C)CC2 N1(C(C(C)Oc2cccc(C)c2)=O)CCCC(NC(=O)CC2CC2(C)C)CCC1 c1(C(N(C(CN(C(C(c2c(C)cccc2)C)=O)C)C)C)=O)ccn2c1CCCC2 C1(c2nnc(-c3sc(OC)c(Br)c3)o2)CCC2COCCC2C1 C(=O)(C(F)CC(C)(C)C)N1CC(C(N(C)CC2CCN(CC)C2)=O)(SC)C1 CC(C)CCC(C)S(=O)(=O)N1CCN(C2(C)CCC2)CC1 CC1CC(CC(=O)NC2(c3ccccn3)CC2)CN1C(c1ncccn1)=O CC(C)C(CNC(C1CCCCO1)=O)C(=O)Nc1cccc2c1OCO2 S(=O)(=O)(c1cc(F)c(F)c(F)c1)N1CC(CNC(c2cc(F)c(F)cc2F)=O)C1 C1(NC(C(CC)OC)=O)CCN(C(C2CCC(=O)N2CC)=O)C1C N1(C(C2(OC)CC2)=O)CCCC(C2CC2NC(c2csc(CO)n2)=O)C1 CN1CCC(CCNC(=O)C(C2CCCCC2)O)C1=O.C12CCCC(C1)C(=O)N2 C1(C(=O)NC(C#C)C(C)OC)C2CCC(C2)N1C(=O)CC1CCC(=O)N1 C1(NC(C(COC)OC)=O)CCC2(CC1)CCN(C(C1(C(C)C)COC1)=O)C2 c1(N2CC(C)(COC)OCC2)nc(=N)[nH]c(=NCC2CSCCS2)[nH]1 C12(CNC(C(CCC)(C)O)=O)CCCC(CN1C(=O)CCNCCCCOC)C2 c1(C(N(CC(C(=O)OC)C)C)=O)cc(CNC(c2ccnc(C)c2)=O)nn1C CC1=C(C(=O)N(C)CCN(C(c2ccnc(OC(C)C)c2F)=O)C(C)C)CCCO1 c1(CNC(c2c(CC)ncs2)=O)ccc(C(=O)NC(C)CC(F)(F)F)cn1 C1(C(=O)NCCC)CCN(C(=O)C(C2CCN(C(C3CCCCC3)=O)C2)C)CC1 C(CO)(C(C)NC(=O)CCSC(F)(F)F)NC(CCOCC(C)C)=O C(=O)(C(C)CCC(C)(C)C)NC(C(=O)N(CCCCCC)CCO)C1CC1 CC1(C)CCC(=CC(=O)NC2CCC(CNC(C3CCCC(F)C3)=O)CC2)CC1 C(C(=O)NCC1(CC(=O)N(C)CC2CCOC2)CC1)(C(C)C)SCC C1(O)(C(C)NC(=O)CC2(O)CCOC2)CCN(C(=O)C2=CCOC2)CC1 c1(C(=O)OC)nsc(=NC2CC(NC(c3ccc(N(C)C)cc3)=O)C23CCC3)[nH]1 C1(C(N(CCNC(CN(C)C(N)=O)=O)C)=O)CCC(O)CN1C C(=O)(CC(CC)CC(F)(F)F)NCC(CC=C)NC(c1cc(C)n(C)c(=O)c1)=O C1(CC)(NC(C2(CC(=O)NC)CCC2)=O)CCN(C(=O)C(C)C(C)COC)CC1 N1(C(c2c(Cl)nc(OC)s2)=O)CCC(NCCC2CCCC2)C(C)C1 C1(CN(C(c2c(CNC(C3(C)CC(=C)C3)=O)occ2)=O)C)CCCC2CC12 N(C1CCCc2cccnc21)(C(=O)C(=O)NCCC(F)(F)F)CCC C=C=CCC(=O)C(=O)C=CC.c1(CN)ncoc1C1CN(C(=O)CCC2CCCCO2)C1 C1(CNC(C2C(C)=CCS2)=O)(NC(=O)CCOCC(F)(F)F)CCCCC1C c1(CC(=O)NC(c2ccccc2F)CNC(c2c(C)con2)=O)ncccc1C C(=O)(CC(C)CC(=O)NCC1CCCCN1C(=O)C(C1CCCCC1)SC)OC C1(CC)CN(C(c2ccc(C)c(Cl)c2)=O)CCC1NC(c1cnc(C(C)C)[nH]1)=O c1(OC)ccc(CNC(N2CCCC(NC(=O)C(C)C)C2)=O)c2ccncc12 C1(NC(CC=C)=O)CC2CCC(C1)N2C(c1cc(-c2ccccn2)[nH]n1)=O C1(C(=O)NC(c2cnn(C)c2)C(=O)N(CC#C)Cc2ccco2)CC2C=CC1C2 Cc1ccc(OCC(=O)NCCC(C(C)C)NC(=O)C(C)CC(N)=O)c(C)c1 C(=O)(C1=C(C)OCCS1)NC1CCC(CCC(=O)N(C(CC)C)C)C1 Cc1nc(C(=O)NC23CCN(C(=O)Cc4cnn(C)c4)CC2C3)c(=O)[nH]c1C C1(NC(CC(CC)C)=O)CCN(Cc2ccn(C)c(=O)c2)CC(C)(C)C1 C1(C)(c2n(CCOC)c(N(CCCN(C)C)C)nn2)CC2(CCC2)C1 C1(CCNC(=O)C(C)=CC2CC2)(OC)CN(C(C2(C)CC2C)=O)C1 CC1(NCc2cn(CCCC3CCCCN3C3CCCC3)nn2)CS(=O)(=O)C1 C1(C(=O)NC(C(C)C)CNC(C2(C(C)C)CCC2)=O)CNC(=O)N1C c1(C(=O)NCC(C)N(C)C(c2ccccc2[N+](=O)[O-])=O)cnn2c1CCCC2 C1(C(=O)NCC2N(C(C3C(NC)C3)=O)CC=C2)CCCN(S(=O)(=O)CC)C1 c1(C(=O)NCCC2CCC(NC(C(C)OCCCC)=O)C2)cc(C2CC2)nn1C C1(N(C(C)=O)CC2CCCO2)CCN(C(=O)C=C2CCN(C)C2)CC1 c1(OC)cc(Cl)c(C)cc1NC(CNS(=O)(=O)NCc1ccccc1Cl)=O N1(C(C2(COC)CC2)=O)C2CCC1C(CNC(c1cc(C(C)(C)C)c[nH]1)=O)C2 Cc1ccnc(C(F)(F)C(=O)NC2C=CC(CNC(c3n[nH]c(C)c3Cl)=O)C2)c1 C1(NC(C(Cc2ccccc2)OC)=O)CC2CCC1N2C(c1occc1C)=O c1(OC)ccc(Cl)c(CN2CC(OC)CC2C(N2CCCC(F)(F)C2)=O)n1 C1(NC(C2(C)ON=C(C)C2)=O)CC2CC(C1)N(C(=O)Cc1cnoc1)C2 c1(CC)noc(C)c1C(N1CCC(CC(C)NC(c2snc(Cl)c2Cl)=O)CC1)=O Cc1[nH]c(=NCCCCC(C)NC(=O)C(c2ccc(Cl)cc2)(C)C)ccc1C#N c1(CN(C(c2cccc(Cl)c2)CCO)C)ccc(C(C)(C)C)cc1 C#Cc1cccc(C(=O)N(CC(C)N(C(=O)CN2C(=O)CN(C)C2=O)C)C)c1 c1(CC(=O)NCC2(O)CC(NC(CC(C)C)=O)C2)cn2ccccc2n1 N1(c2cccc(N(C)C)c2)C(=O)CC(Nc2nc(-c3nn[nH]n3)c(Cl)s2)C1=O C1(C(N(C)CCn2cncn2)=O)CCC2(CC2)N1C(C1(C#N)CC1(C)C)=O C#CCC(C(=O)N1CCC1(C)CC(=O)NCC(CO)N(C)C)C1CC1 N1(C(C=CCOC)=O)CC(CNC(C2COC(C)(C)C2)=O)C(C)C1 c1(OC)ncccc1CCC(=O)N(C1CCN(C(C2CNC(=O)C2)=O)C1)C N1(C(c2ccc(C#C)cn2)=O)C2CCC1CN(C(c1nccn1C(C)C)=O)C2 Cc1cocc1C(N1CC=CC1CNC(c1ncsc1-c1ccccc1)=O)=O c1(C(=O)NCC(CC)(CC)NC(c2ccoc2Cl)=O)ccc(C(F)(F)F)nc1C CC1CC(NC(=O)NC2CC3CCC(C2)O3)CCN1C C1(CNC(CCCC=C)=O)CCN(C(=O)C(=C2CCCCC2)F)CC1C c1(C(=O)NC2CC(N(C(c3c(CC)n(C)nn3)=O)C)C2)nc(O)nc(O)c1N C#CCC(C(=O)N1CC(c2ncc[nH]2)C1)NC(c1ncncc1Cl)=O C(C(F)(C(=O)N(CC(Cl)Cl)C)C(C)C)NC(c1c(CC)ocn1)=O CC1=C(C(=O)N2CCN(C(=O)C(C)Cc3cnn(C)c3)CC2C2CCC2)CCC1 c1(Cc2ccc(CNC(C3(S(C)(=O)=O)CCC3)=O)cc2)nnc2ccccn12 c1(-c2ccc(C(=O)NC(CCC)CO)nc2)ccc(S(=O)(=O)N2CCSC2)cc1 c1(C(=O)Nc2ccc(NCCn3cc(Br)ccc3=O)cc2)cccc2c[nH]nc12 N1(c2nc(C)nc(=N)[nH]2)CCCC2(NC(C3CCS(=O)(=O)N3)=O)CC2C1 c1(C(=O)NCC(C)NC(C(C)OCC)=O)ccnc(-c2ccccc2)c1[N+](=O)[O-] c1(OC)nc(C)cnc1C(=O)NCC1(NC(=O)CC2C=NN(C)C2=O)CCCC1 N(C(=NCCF)NC1CCCc2nc(C)sc21)CC1C(=C)C1 N1(C(CN2CC(C)(OC)C2)=O)CCN(C(c2cc3ccsc3s2)=O)C(CO)C1 C1(NC(C2CN=C3N=CNN3C2)=O)CN(C(=O)CSC2CC2)CC2CCCC12 c1(N(C(C)COC(F)F)C)nc(=NC2CC2C)[nH]c2c1COC2 C1(C(N(C)Cc2nccs2)=O)CN(C(=O)C(F)CC2CCOC2)CC1F N1(C(C(CNC(C=C(CC)CC)=O)C)=O)CC2(CC(OCC)C2)C1 c1(C(C)C(=O)NC(C(=O)NCC(F)(F)F)C2CCOC2)ccn(C)c1 c1(NC(C2CC2CNC(C2COCCO2)=O)=O)ccc(-c2ccccc2)nn1 N1(S(CC2CCC2)(=O)=O)CC(NC2C(C(=O)OC)C2)CC1C CC(C)C(C#N)C(=O)NC1C(C(=O)NCC2(n3cccn3)CC2)C1(C)C Cc1nn(C)c2c(N(C)Cc3sccc3Br)nc(N3CCCC(C(C)C)C3)nc12 c1(C(N2C(CNC(C3N(CC)CCC3)=O)CC2)=O)cnn2c1CCCC2 c1(OCC2(NC(C3CN(c4n(C)nnn4)C3)=O)CCC2)ccccc1Br CC1(NC(c2coc(CC3CC3)n2)=O)CCCN(C(C2(F)CCCCCC2)=O)C1 N1(C(C2(CC)CCCO2)=O)CC2=C(C1)CN(C(=O)CCOc1ccccc1Cl)C2 C1(NC(CCNC(=O)OCC)=O)CCCC2CN(C(C3CC(F)(F)CS3)=O)CC12 C1(CC(C)NC(=O)CC2C=CCCC2)CCN(C(=O)Cc2nncn2C)CC1 c1(CNC(CNC(c2c(C)occ2)=O)=O)ccc(CNC(=O)CCCC#N)cc1 CCCC(C(O)C(=O)NC1CCN(C(C)C)C1)NC(=O)CC1CCSCC1 c1(CC)cccc(NC(=O)C(CCNC(C2CC(C)N(C)C2)=O)OC)c1 c1(C(CC(=O)O)NC(CC2(C(=O)OC)CC2)=O)cc(C)c(F)cc1F C1(NC(C2CCOCC2)=O)CN(C(=O)CN2CCSCC2)CC1n1ccnn1 N1(C(C(=O)NCC)=O)CCCC1C1CCCN1C(c1cc(=O)c(OC)cn1C)=O c1(C(N2CC(C)CN(C(=O)CC(C)C3CC3)CC2)=O)ccc2c(c1)COC2=O C1(NC(CCSC)=O)CCN(C(=O)CN2CCOCC2)C1C1CC1 C=C(C)C(C)(C)C(=O)NCC1(O)CC(NC(c2cc(Cl)ccn2)=O)C1 C1(ONC(CNC(CNC(CCCSC)=O)=O)=O)COC(C)(C)C1 C=CCCCC(C(=O)N(C(CF)CF)C)NC(C1CSC1)=O C1(NC(C(C)NC(CC)=O)=O)CCCCCN(C(=O)CC2CCCCCC2)C1 c1(OC)ccc(CC(=O)NC(C)C(c2ccc(Cl)cc2)O)cc1[N+](=O)[O-] N1(C(c2nc(OCC)oc2)=O)CCC(C2CCCN(CC(C)O)C2)CC1 c1(C(=O)NCC(CN(C(Cn2c(C)nnn2)=O)C)O)cc(C(F)(F)F)ccc1Cl CCCC(CC)CCC(=O)N1CCCC(NC(=O)CCC(C)C)C1 Cc1cc(C(=O)NCC(C(C)C)NC(=O)C(C)(C)C2CCOC2)oc1C C1(OC)CN(C(C2CCOC2(C)C)=O)CC1C(N1CC(CO)C(O)C1)=O c1(C(=O)NCC2N(C(C(CC)CC)=O)CC2)cnn2c1CCCC2C C1(C(c2nnnn2-c2ccc(F)cc2)NCC(C)F)CCC2CC1C2(C)C c1(C(=O)NCC(C)N(C(=O)C=Cc2nccnc2C)CC)cc(C)cc(C#N)c1 O=C(NNc1ccc(Cl)c(-c2nn[nH]n2)c1)C1COc2ccc(OCC(F)F)cc21 N1(C(CC2N(C(C3=C(C)CCC3)=O)CCCC2)=O)CCCNC(=O)C1C(C)C Cc1ccc(Cl)c(OC(C)C(=O)NC2CCCN(C(=O)CC3(CO)CC3)C2C)c1 c1(C(N(C(CC)CC(=O)NCC(c2nncn2C)C)C)=O)ccc(N)c(F)n1 Cc1cscc1C(=O)NCCNC(=O)CSCC(c1ccccc1)=O C(=O)(CC(=O)NCC1CCC(NC(c2[nH]nnc2C)=O)C1)NCC#C c1(C(N2C3C(CNC(c4cccnn4)=O)C(C3)C2)=O)ccc(Br)c(Cl)c1 C(C(=O)NC1CC1NC(=O)Cc1ccc(F)cc1F)(C(C)(C)C)NC(C)=O C(C(C)CC(=O)N1CCC(C)(C(=O)NCC2CCC2(F)F)C1)OC c1(NC(CCCCC)c2nnnn2C2CC2)cc(Cl)cc(Br)c1 c1(C(=O)NCC(C)NC(C=CC(CC)C)=O)ccc(OCC(C)C)nc1 C(CCCCC(=O)NC(C1CCOCC1)C)NC(CC(C)CN(C)C)=O Cc1nnc2n1CCN(C(C1C=CC(NCc3ccsc3Br)C1)=O)C2 C1(CSC)CCN(C(c2cc(C(=O)OC)cs2)C(=O)NC2COC2)CC1 C1(O)(CNC(=O)Cn2ccccc2=O)CCCN(C(c2cc[nH]c2)=O)CC1 C(c1ccc2c(c1)COCC2)=CC(=O)NC1(C)CN(C(CN2C(C)CCC2)=O)C1 C1(C(=O)NC(CC)C)CCC(C(C)C)N1C(=O)CC1(OC)CCC1 C1(NC(c2c(C)scc2)=O)CN(C(c2c(Br)nnn2C)=O)CCC1CO C(C(C(C)(C)C)NC(=O)CC1(C)CCCCC1)NC(CN(C)C(=O)C1CC1)=O c1(CNC(=O)NC2C3CN(CC)CC2CC3)cccc2c1nnn2C c1(NCOC(COC2C(C(C)C)CCCC2)=O)cc2cc(Br)cnc2o1 c1(CC(=O)OCCOC(C(c2ccc(OC)cc2)=O)C)cccc(Br)c1Cl C(C(CO)C(F)(F)F)Sc1cccc(C(F)(F)F)c1.O=C1CCCc2c[nH]c(c2)N1 C1(NC(C(C)(C)NC(=O)OC)=O)CCOCC1C(=O)NCCC(O)C1CCCC1 C(=O)(C1CCCn2ccnc21)N1CCC2CN(C(c3ccc(C)c(C)n3)=O)CC21 C1(CNC(CN2CC(C)(OC)C2)=O)(CNC(=O)Cc2cn[nH]c2)CC2CCCC2C1 C1(NC(C(Cn2ccc(C)n2)C)=O)CCCCN(C(C2CCCC(=O)C2)=O)C1 C1(COC)(CNC(C2CCC2)=O)CCCN1C(C1CCSCC1)=O C(C)(CC(C)N=c1nc(C)cc(C)[nH]1)NC(CCCCCC=C)=O c1(SC)cc(C)ccc1C(N1CC(N(C(=O)CC(C)F)C)C2(CC2)C1)=O CC(Cc1cnc[nH]1)C(=O)N1CC(CC(=O)NCCOc2ccncc2)C1 N1(C(=O)Nc2cccc(C)c2Cl)CCCC2(CNC(=O)C2)C1 c1(NC(c2cc(C(F)(F)F)cc(F)c2)=O)ncc(Br)nc1Cl.C12CC1CNC2=O CC(O)C(F)(F)C(=O)NCCCOCCOCCNC(=O)CC1CCC=CCC1 C1(CC)CCN(C(C2COCCN2NC(C2CC23CNC3)=O)=O)CC1 C1(S(C)(=O)=O)(C(=O)NCC2C(NC(c3ccc(C)c(F)c3N)=O)C2)CCOCC1 c1(CC)ccc(C(N2CC(O)(C(C)NC(=O)C(C)CCN(C)C)C2)=O)c(F)c1 c1(CC)ccc2c(Cl)c(C(=O)NC3(C)C4CCCCC34)sc2c1 Cc1c(Cl)ccnc1C(N1CCCC(CNC(=O)C2=NOCC2)CC1)=O C1(N(C(c2c(C)scn2)=O)C)CN(C(=O)CCc2cccc(C(F)F)c2)CC1F C12(C(=O)OC(C3CCN(C(CCC(=C)C)=O)C3C)=O)CC3CC(CC(C3)O1)C2 C(C(CC=C)C(=O)NCC1(F)CC(CO)C1)NC(C(CC#C)O)=O N1(C(c2c(CC)onc2)=O)CCN(C(c2oc(C3CCC3)nc2C)=O)CCC1C c1(OCC)ccc2cc(-c3ccc(C(O)C(=O)OCC4CCC4)cc3)ccc2n1 C1(NC(C2N(CCC)CCCC2)=O)CCN(C(=O)C(C2CCCCC2)O)CC1F CCC(C)(CC)C(=O)NC(CNC(c1cccc(-c2ccncc2)n1)=O)CO CC(C(=O)NNC(=O)COC(=O)COCc1nc[nH]n1)C1CC1 C(=O)(CC1=NNC(=O)C1)NC1CN(C(C(=O)NC)(COC)NC(=O)C(C)(C)C)CC1(C)C c1(COC)cnn(-c2ccc(C)cc2)c1C(N1CC(O)C1)=O.C12CCC(C1)N2 c1(OC)ccc(C(=O)NCC2(C)CCCN(C(c3ccon3)=O)C2)c(OC)c1 O(NC(=O)CC(C)(C)C)C(C(=O)NCCC(C=C)C)CC(C)C c1(C(=O)NC(CC)CNC(=O)Cn2ncccc2=O)ccc2c(c1)OCCN2 C1(CC)(NC(=O)Cc2cccn2C)CCN(C(=O)CN(C(=O)C(C)C)C)CC1 C12CCN(CC1)Cc1cn2nn1.c1(C(=O)NC2(CCC)CC2)ccn(CC)n1 CC(CN=c1cccc(S(=O)(=O)NCCC23CCC(CC2)OC3)[nH]1)C(F)(F)F C(C)(COC)(CCO)NC(CSCCNC(CSCC=C)=O)=O NC(=O)CCC(=O)NCCC1CCCN1C(C1SCCCS1)=O C1(C(=O)NCCCCn2cc(C3CCOCC3)nn2)Cc2ccccc2NC1=O C1(C(=O)NCC(C(C)C)(C)NC(=O)CCc2ccc(O)nc2)CCC(F)(F)CO1 C=CC(CC)CC(=O)NC(C1CCCN1C(c1cc(-c2cnn(C)c2)on1)=O)C N1(C(c2nc(NC(C)=O)sc2)=O)CCC(NC(C2(C)CCCC2O)=O)C1C Cc1ccc(F)c2c1CCN(Cc1cn(CCC3CCNCC3)nn1)C2 c1(OC)cc(CC(N2C3CCC2(CNC(c2cncs2)=O)CC3)=O)ccc1O C1(NC(c2ncn(C)n2)=O)CCN(C(c2cc(C(F)(F)F)ncc2Cl)=O)CC1F CCCCC(C(=O)NC1CCC(F)(CNC(C2(S(N)(=O)=O)CCC2)=O)C1)C(C)C n1(CC(C(=O)OCC)O)cc(C#CCNC(=O)C2=CCCO2)nn1 C1(NC(CNS(CC)(=O)=O)=O)CC(C2CCN(C(=O)CCN(C)C(C)=O)C2)C1 Cc1nn(CC(F)(F)F)cc1C(=O)NC(C)CNC(C1(C)CC2CC2C1)=O c1(C(=O)NC2C=CCN(C(CCC3OCC(C)(C)C3)=O)C2)ccc2snnc2c1 c1(C(=O)NC2(Cc3ccccc3)CC23CCC3)cccc2c1OCO2 N1(C(c2n(CC)ncc2)=O)CCCC(C(=O)NCCCC(=O)OC)C1 C1(NC(C2N(C)C(=O)CC2)=O)C2CC3C(C2)C13C(=O)NN1CC(CO)C1 C(=O)(CC(C)P(C)(C)=O)N1CCC(F)(CNC(C(C)OCCCC)=O)CC1 C=CCC(CC=C)C(=O)NCC(C)CN(C(=O)Cc1cccc2sccc12)C C1(NC(C(CC)(F)F)=O)CN(C(C2CC23CCOCC3)=O)CC2(CC2)C1 Cc1c(C(N2CCCC(CN(C(=O)C3=NNC(=O)C3)C)C2)=O)[nH]c2c1CCCC2 CC1(C)Oc2ccc(NC(C3CCN3Cc3c(O)ccc(F)c3Br)=O)cc2O1 C12(NC(c3nnn(CC)c3C)=O)CCC(C(N3CC(O)(CC(C)C)C3)=O)(CC1)C2 C1(C(=O)NCC2CC[Si](C)(C)C2)CC2CCCC2N1C(=O)C(=O)C1CCCC1 C1(CNC(c2cccc(CC)n2)=O)C(C2CC2)CCN1C(=O)C(F)OC Cc1nc(C)c(C(=O)NCC2(C)CCN(C(=O)C(c3ccccc3)F)C2)[nH]1 C12(CNC(c3c(C(C)C)occ3)=O)CC(CO1)N(C(C1CC(=O)NC1(C)C)=O)C2 c1(NC(C2CCCN2C(=O)Nc2ccsc2)=O)ccccc1OCC1CC1 C(C(C(=O)NC(CC1CCCC1)C(=O)O)N(C)C)NC(C)=O C(=O)(C1=CC2CCCC12)NC(C1CCCCN1C(C1CC2CC2C1)=O)C C1(C)(C(=O)NCC(CC)NC(C2CN(C3CCN(C)CC3)C2)=O)CCCCC1 c1(C(=O)NCC2C(NC(c3c[nH]c(Br)c3)=O)C2)scnc1Cl N1(C(C2CCCN(C(C)=O)C2)=O)CCN(C(c2ncn(C)n2)=O)CC1CC1CC1 N(C1CCn2ccnc21)C(c1ccc(NCc2cncs2)cc1)=O O=C(CCCC(F)F)N1CC(CN2CCN(C(=O)CC3CC4CCC3O4)CC2)C1 c1(C(=O)NCC(CNC(c2cc(Cl)cc(Cl)n2)=O)O)ccnc2[nH]ncc12 c1(CN(C(COC)C)Cc2sncc2C)ccc(Cl)cc1 N1(C(C(COC)(C)C)=O)CC2CCC(NC3CN(C(=O)OC(C)(C)C)C3)(C2)C1 Cc1ccc(CN(C(c2sccc2Cl)C(=O)NC2CCC2)CC(C)C)o1 c1(C(=O)Nc2c(OC)cc(C)cc2)ccc2nc(-c3ccsc3C#N)cn2c1 C1(NC(C(N2CCC(O)CC2)C)=O)CCC(C)N(C(C2CSCC(=O)N2)=O)C1 c1(C(=O)NCC2(NC(C(C)=C(CC)C)=O)CC2)nccc2nn[nH]c12 C=C1CC(C(=O)NCC(C)(CNC(C2CC2CC)=O)OC)(C(F)F)C1 c1(OC)cc(N2CCCC(CCNC(=O)CCC3NC(=O)NC3=O)C2)ncn1 CC1CC(=O)NC1C(=O)NCC1CCC(NC(c2cc(O)no2)=O)C1 C(=O)(CC1OCc2ccccc21)N1CC=CC(NC(C23CCC(C)(OC2)C3)=O)C1 C1(NC(C2CCC(=C(F)F)CC2)=O)CC12CCS(=O)(=O)CC2 c1(CCC(=O)NC(CNC(C=C(C)C(F)F)=O)C)cnc(O)[nH]1 N#Cc1ccc(=NC2CC2C(N2CCC(C3(O)CCC3)CC2)=O)[nH]c1 C1(C(=O)NC2(C#N)CCC2)CC12CCN(C(c1ccc3ncsc3c1)=O)CC2 CC(C1CCCCC1)=CC(=O)NC1(C)CCN(C(C2(C)CCCCO2)=O)CC1 N1(C(CC(C)(C)C)=O)CC(F)(F)CC1CNC(c1nsnc1O)=O Cc1nc(CC(=O)NCC(C)(C)OCCNC(c2cc(CF)on2)=O)n[nH]1 C(=O)(C1=C(Cl)CCC1)N1CC(C(C(=O)N(C)CCc2cnn(C)c2)O)C1 c1(C(=O)NCCCNC(CC2C(C)(C)CCO2)=O)cccc(N=S(C)(C)=O)c1 N(C1CCCOc2c1ccc(Cl)c2Cl)C(=O)NC1CC2CCC1O2 C=CCCC(=O)COC(=O)CSCCc1c(C)noc1C CCCCC(F)C(=O)NC1CCN(C(C2CCS(=O)(=O)N2)=O)C(C)C1 CC1CCC(CNC(=O)CC2(NC(C)=O)CC2)CN1C(=O)CCS(N)(=O)=O N1(C(C(C)CS(C)=O)=O)CCc2c(c(CNC(c3nnc(S)n3C)=O)nn2C)C1 C1(C(N2CC(N(C(C=Cc3cnc(C)s3)=O)C)C2)=O)C2(CC2)C12CC2 C(C(C)(C)C(=O)NCCC1CN(C(=O)C(c2ccc(C(C)C)cc2)(C)C)C1)OC CCC(CCCC(=O)NC(c1ccns1)C)NC(C1(OC)CCOC1)=O C1(NC(c2cncc(F)c2)=O)CN(C(=O)Cn2cc(Cl)cn2)CCC1C(F)(F)F Cc1cc(F)cc(Br)c1NC(N1CCC(COCC2CC2)CC1)=O N1(C(C2CCN(CC)C2)=O)CC(NC(C2CN(CC(F)(F)F)C2)=O)C(SC)C1 C=CCN(CCOc1ccc(OC)c(Cl)c1)N1CCOCC1C(C)C CC1CC2(CO1)CN(C(C1(NC(=O)CC3CCSCC3)CCOCC1)=O)C2 N1(CCc2cn(Cc3ncc(C)o3)nn2)CCCN(C(=O)Cn2ccnn2)CC1 c1(C(N(CCC(C)NC(=O)C=CC2CCC2)C)=O)ccn2c1CCCC2 c1(C(=O)NC2(C#N)CCN(C(c3c(C)ccnc3)=O)C2)cc(F)c(F)cc1I N1(C(CN(C)C2CC2)=O)CCC2(CC2NC(=O)CC2NC(=O)NC2=O)C1 C1(C(=O)NCC(CN(C(c2c(CC)ocn2)=O)C)(C)C)COCCC1(F)F C1(NC(C2CCCCN2C(=O)CCC2CCCOC2)=O)CC2(CCOC2)C1 C1(O)(CNC(C(C)(C)NC(c2nnn(CC)c2C)=O)=O)CCCC(C)C1 C1(CNC(C(CCC)CC)=O)CN(C(C2(OC(C)C)CCC2)=O)CCC12CCC2 c1(OCCOC)ccc(C2CC2NC(=O)NCCS(=O)CC)cc1 C(C)(CC(C)(C)OC)NC(C(COC)Oc1ccccc1)=O C1(C)(NC(C(c2cnn(C)c2)NC(c2ccc(CC)[nH]2)=O)=O)CCC(O)CC1 N1(C(CC(=C)C)=O)CCC2(CCCCN(C(c3cnc(N(C)C)nc3)=O)C2)C1 C(=O)(CCC(C)(C)N(C)C)N(C1CCN(C(=O)COCCC(C)C)CC1)CC#C C(CC)(CCC(=O)NC1C=CCC1)NC(CNC(CCC)=O)=O C1(NC(C2C(C)C2)=O)CCCC12CN(C(c1cnn3c1OCC3)=O)C2 N1(C(CCc2cccc(OC)n2)=O)CC2CCCC(C1)N2C(C1CCCOC1)=O C(=O)(CC(C(F)F)n1ccnc1)N(C(C)C)CCNC(c1[nH]nnc1C1CC1)=O Cc1oc(CNC(=O)CC2CCC(C)O2)nc1C(=O)N(C)CCOCC1CC1 N1(C(c2nc(C(=O)NC(C)=O)sc2)=O)CCN(CCNC(=O)CC2(C)CC2)CC1 Cc1nn2cc(CC(N3CCC(C#N)(NC(=O)CCc4ccco4)C3)=O)nc2s1 Cc1oc(Br)cc1C(=O)NC1CCN(C(c2nn(C)cc2N)=O)C1C(C)(C)C C1(C(=O)N(C)CC2CCC2)(CC)CCN(C(C2CCCCC2C)=O)CC1 c1(CCC)[nH]nc(C(=O)N(C2CC(NC(C3CSCC(=O)N3)=O)C2)C)c1[N+](=O)[O-] c1(OCC)cc(C)ccc1Oc1cc(-c2cnn(C)c2)ncn1 c1(C(=O)NCC#CCNC(C(C)OC)=O)cc(NC(C)=O)cnc1C N1(C(c2coc(Cl)n2)=O)CCC2C(CCCN2C(c2[nH]nc3ncccc23)=O)C1 C1(NC(CSCCC)=O)C2CCN(C(c3cn(-c4ccccc4)nn3)=O)CCC12 Cc1cc(NC(=O)CN2CCC(C(C)(C)O)C2)ccc1F S(=O)(=O)(c1ccc(OC(F)(F)F)c(Br)c1)NCCOC(c1cc(C)cc(C)c1)C(=O)O N1(C(c2ccc(C#C)s2)=O)CCC2(NC(=O)CCOc3ccc(F)cc3)CC2C1 N1(C(c2cc(C)nc(C)c2)=O)CC2(CNC(C3CCS(=O)(=O)C3)=O)CC(F)(C1)C2 NC(=O)CCC(C(=O)N(CC(O)Cc1ccc(Br)cc1)C)n1ccnc1 C1(C(N2CCN(C(C)C(=O)Nc3cncc(Br)c3)CC2)=O)CCC2(CCC2)CC1 C1(C(N(CCCn2cc(CCCCCCO)nn2)C)=O)CCCCC12CC2(F)F c1(C(N2CC3N(C(Cc4c(C)n[nH]c4)=O)C(C3)C2)=O)ccn2ccnc2c1 Cc1cc(C(=O)NCCC2CCCN2C(C23CCC(CO2)C3)=O)c(Br)c(C)c1 C(=O)(C=C=C(C)C)N1CCC(CCC(=O)NCC(C(=O)OC)O)C1 C1(NC(C(CC)N(C)C)=O)CCC(C)N(C(c2nnn(C(C)C)c2C)=O)C1 C12(CNC(=O)C(F)C3CCC3)CC(CO1)N(C(=O)C=CSc1ccccc1)C2 c1(C(=O)NCC(CNC(CCCOCCOCC)=O)F)c(N)cc(Cl)cc1F c1(-c2cccc(C(N(CCC#C)C)=O)c2)cc(C)nc2ccnn12 N1(C(CCN(CCC(C)(C)C)C)=O)CCCC(n2cc(CCS(C)(=O)=O)nn2)C1 c1(C(=O)OC)cc(COC)cc(S(=O)(=O)NC2CCC(c3ccccc3Cl)C2)c1 C1(C(=O)NCC(CCNC(CNC(=O)OCC)=O)O)CCCCN1C c1(CC)nn[nH]c1C(=O)NCc1cn(CCNC(c2cc(C)[nH]n2)=O)nn1 CC1CCN(C(C2CCS(=O)(=O)N2)=O)CC1NC(c1occc1C1CC1)=O N1(C(COC2(C)CN(C(C3CC(C)N(C)C3)=O)C2)=O)CC2(CCC2O)C1 Cc1ccnc(C)c1CNC(C1CCN(C(=O)Cn2ncccc2=O)CC1C)=O N1(C(C2CC(F)(CF)C2)=O)CCN(C(C2CCCCS2)=O)C(CO)C1 CC1(C)CCCOC1C(N1CCN(C(C2CCC2)=O)CC1CCO)=O C12(C)CCCC1NC(=O)C1(CCSC1)NC2.C1(CC(=O)OC)COCCOC1 c1(C(N2CC(CC(C)O)C2)=O)cccc(-n2cc(CC(C3CCCC3)N)nn2)c1 C=C(C)CCCC(=O)N1CCC(C)C(CNC(=O)CCNC(c2ccco2)=O)C1 c1(C(=O)NC2C=CC(CNC(COCC)=O)C2)cn2ncccc2n1 c1(C(N2CCC3(NC(=O)CCCCC4CC4)C(C2)C3)=O)ccc2nccn2n1 N1(C(CCC)=O)CCN(C(=O)C(CCSC)NC(c2cn(CCO)nn2)=O)CC1 C1(C(=O)NCc2ccc3nc(C)sc3c2)CC(O)c2ccccc2O1 Cc1cc(C(N2CCC(C(N)=O)C23CC3)=O)ncc1CNC(=O)C(C)SC(C)C N1(C(CCOCC)=O)CCOCC(NC(C2CC(=O)N(C(CC)CC)C2)=O)C1 c1(NCc2c(C)cccc2)cc(N2CCC(OCC(F)F)CC2)nc(C(C)C)n1 C12(NC(C=CCC)=O)CCCN(C(c3ccc(OC)cc3N)=O)CC1C2 C=C(Cl)CC(C(=O)NCCN1CCOCC1=O)NC(=O)CCn1cccn1 C1(N(CC#C)C(C2CCN(C(=O)CC3(C)CC3)C2)=O)CCN(C(=O)C(C)C)CC1 C1(CCC(N2CCC(n3ccnc3)C2)=O)CCCCN1C(=O)Cn1cccc1 CC(C(=O)N1CC(OCCN(C(=O)COCC(C)(C)C)C)C1)C(C)n1cccn1 CCC(CC)C(C)C(=O)NCC1CCCCN1C(=O)CCc1cccnc1Cl c1(C(=O)OC(C)C(=O)NC2CCCCC2)cccc2c1SCCC2=O n1(C(C)C)ncc2c(N3CCC3C(=O)NCCOc3cccc(Cl)c3)ncnc12 C1(C(N(C)Cc2ccn(CC)n2)=O)CC2(CCN1C(c1ccsc1C)=O)CC2 N1(C(c2ccc(C)s2)=O)C2CCCC1CC(NC(C1(c3cc[nH]n3)CC1)=O)C2 Cc1nc2cnn(C)c2cc1C(=O)NC(C)CNC(=O)CCN1CCCCCC1 c1(C(=O)NC=C(C=CC=C)C)cc(C)n(CCNC(=O)OC(C)(C)C)c1C N1(C(C2N(C(C(C=C=C)C)=O)CC3CC32)=O)CCc2nocc2C1 c1(C(=O)NCCCN(C(c2cc(C)c(C#N)cn2)=O)C)sc2cccnc2c1Cl C(=O)(CC(C)C(=O)N1CC(N(C(=O)CC2CCC2C)C)C2(CC2)C1)OC CC1(CNC(=O)Cc2cc(O)nc(O)n2)COCCN(C(C2CC2C2CC2)=O)C1 c1(CC(=O)NC2C(NC(C(C)NC(N)=O)=O)C2)cc2ccccc2c(O)n1 C12(C(N3C(C)(CNC(C4CC(=C)C4)=O)CCC3)=O)CCCC1C2(F)F C12(C(N3CCC(C(=O)NC4CN(C(C)=O)C4)CC3)=O)CC3CC(CC(C3)C1)C2 N1(SC)CCCN(C(=O)NCc2cccc(NC(=O)OC(C)(C)C)c2F)CC1 C1(C)(CNC(CNC(=O)NC)=O)CCCN1C(c1nn[nH]c1Cl)=O c1(C(N2C(C)C(NC(C3C4CCCC34)=O)CC2)=O)cccc(F)c1O c1(C(=O)NC(C(C)(C)NC(Cc2cc(C(=O)OC)sc2)=O)C)cc(C)cc(O)n1 n1(CC)cc(Br)c(CC(N2CCCC(CC3CCCCC3)C2)=O)n1 Cc1c(NC(C2(CNC(=O)C(C)(C)C)CC2)=O)cc(F)cc1Br C1(C(=O)NCCCC2N(C(c3ccn(CC)n3)=O)CCCC2)CCOC(C)(C)C1 C1(CNC(CN2CC(CC)C2)=O)(CNC(c2c[nH]nc2C2CC2)=O)CCCC1 N1(C(C(CC)OC2CCCC2)=O)CCC(C)(NC(=O)Cc2csnc2C)CC1 C(=O)(C1=CCC(F)(F)CC1)N1CCN(C(=O)CCN2CCCC2)C2C1C2 C1(CNC(C2CC(CN(C)C)C2)=O)CC2(CC2)CN1C(=O)Cn1c(C)ccc1C c1(NC(=O)NCCCOCC(F)F)ccccc1F C1(C(N2C(CNC(C=C(CC)C)=O)COCC2)=O)CC2(CCC2OC)C1 N1(C(C2CN(CCC)C(=O)C2)=O)CC(C2CCCCN(C(c3ccon3)=O)C2)C1 C1(CC(=O)NCCC2CCN(C(C3CC(F)(F)CS3)=O)C2)CCC(=O)NC1 c1(C(=O)NCC2C(NC(C3(OC(C)C)CCC3)=O)CCC2)ocnc1C(F)(F)F c12cc(ccn1)CCCNC(=O)CNC2=O.CC1CCC(CO)C1 c1(OCC)ccc(C)cc1NC(C)C(=O)Nc1ccc(Cl)cc1 c1(OC)ccc(CN2CC(C)(C(=O)NCC3CCCCO3)C2)c(Cl)c1O C12(NC(c3cn(C)c(C(F)F)n3)=O)CCC(COCCO)(CC1)C2 C(=O)(C1CCCc2nncn21)NC(CC(C)NC(CC1(OC)CC1)=O)C C(C#CC1CC1)NC(=O)CCNC(C1CCSCC1)=O N1(C(C2C(C)C2C)=O)CCCC2C1CCN2C(c1ccc(C#N)cc1O)=O C(=O)(CN=c1cc[nH]cc1)N1CCC(C(=O)NCC(C)OC)C1(C)C C1(C(=O)NCCCCC(=O)NCC(C)(C)n2cccn2)CC2CC1CC2O C(C)(C(CO)NC(=O)CCCNC(C)=O)NC(C(C)NC(CC)=O)=O C=CCCC(CC(C)C)C(=O)NCC(C1CCCCC1)NC(=O)CCOC(C)C C1(CC)CCCN(C(=O)Cc2cc(C)no2)C1C(=O)NCC1CC1 N1(C(c2c(OC)scc2)=O)CCCCC(NC(c2nnc(C(C)(C)C)s2)=O)C1 c1(C(=O)NC2C(NC(C3(CC=C)CCC3)=O)C2)cc(Br)cn1C(C)C CC1CC(C(=O)NCC2(CNC(c3cn4ccsc4n3)=O)CC2)CC(C)C1 n1(CC)c(O)nc2cc(C(N3CCC(NC(=O)CC(C)CF)CC3C)=O)ccc12 CC(C)(C(=O)NCC1CC(NC(=O)C(F)(F)C(O)C2CC2)C(O)C1)S(C)(=O)=O C1(C(NOCCOCCOC)=O)(C(C)C)CCCN1C(c1oc(C)nc1C)=O Cc1oc(C)c(C(N2CCC(C)(NC(c3cc(O)cc(O)n3)=O)C2)=O)c1C CC(O)C(C)NC(=O)C(C1CC1)N(C)C(C1CC(=C2CCC2)C1)=O C1(C(=O)NCC(C)(C2CC2)NC(CCN(C)CC)=O)CC2(CCO1)CC2 C1(O)(CN(C)C(c2scnc2Cl)=O)CCN(C(=O)CC2CCC3(CCC3)O2)CC1 c1(C(C(=O)NCC(C)NC(=O)CNC(=O)C2CC2)C)ccc(Cl)cc1 C(=O)(C(O)CCC(F)(F)F)N1CC2(C(NC(C3CSCCS3)=O)CCC2)C1 C(=O)(C1=CCCCC1)NC1CC1.C12CCN(CC1)Cc1cc(on1)C(=O)NC2C N1(C(C(C2CCN(C(c3c(C)ccnc3C)=O)C2)F)=O)CCCN(C)CC1C N1(C(C=CC(C)=O)=O)CC(NC(=O)Cc2nccn2C)CC1C C(C(=O)NC1CCCN(C(c2conc2C)=O)C1C)(C(C)(C)C)SC N1(C(c2c(COC)cco2)=O)CCCC(NC(=O)CN(S(C)(=O)=O)C)CC1 c1(C(=O)NC2C(CNC(c3c(C)n[nH]c3)=O)C2)cc(Br)cc(C(F)(F)F)c1N N1(C(C(N)=O)=O)CCc2sccc2C1CNC(c1cc2c(O)cccc2[nH]1)=O C(C1=CCN(C(C2(F)CCN(C(=O)CC(C)C3CC3)C2)=O)CC1)OC C1(CNC(c2nn(CC)c(C)c2)=O)CC(C)(C)CN1C(c1[nH]ccc1COC)=O c1(SCC(N2CCCN(C(C3C(OC)CCC3)=O)CC2)=O)ncnc2[nH]cnc12 C1(NC(C2CN(C(C(C)SCCCC)=O)CC23CC3)=O)CCC2(CCCC2)C1 C(=O)(CC=C(Cl)Cl)NC(C)CC1CN(C(=O)CN(c2cnccn2)CCO)C1 Cc1cc(CN=C(NCc2ccco2)NC2CC2C(F)F)c(C)o1 C1(C(=O)NCC2C(C)CCC2)C2CC1N(C(c1ccc(O)nn1)=O)C2 Cc1nsc(C(=O)NC2(C(=O)NC(CO)CCCO)CC2C)c1N CC1CC(=O)NC(C(N2CC(OCC(=O)N(CC(O)C(C)(C)C)CCO)C2)=O)C1 CC1CN(C(=O)CCC2CC2C)CC1(C)C(=O)N(C1CC2CCC1CC2)C C1(CC)(NC(=O)CCCC2CC2)CCCN(C(c2c[nH]nc2C2CCOC2)=O)C1 c1(N2CCOCC(CNC(CN(C3CCC3)C)=O)C2)c(Br)cncc1[N+](=O)[O-] C1(C(CNC(COCC(=O)NC)=O)O)CCN(C(=O)C(C(C)C)NS(C)(=O)=O)CC1 C1(C)(CNC(CCCOC(C)=O)=O)CCN(C(c2ncnc(O)c2F)=O)CC1 c1(OCC)ccc(NC(=O)NCC2(OCCOC)CCCC2)c2cnccc12 c1(CNC(C2N(C(c3cc(C)n(C)n3)=O)CC(O)C2)=O)c(F)cncc1F N1(C(C=CCCC)=O)CCN(C(=O)C(n2ccnc2C)C)C(CCO)C1 CC1CCC(C(=O)NC2COCC2O)N1C(c1cnc[nH]1)=O c1(OC)c(CN(c2cc(NCC(Br)=C(C)C)ncn2)C)cccc1Cl C1(C(=O)NC(CNC(C(C=C)(C)C)=O)CC)CCC(=O)N(CC)C1 O(NC(=O)C(CNC(=O)CCCC(F)(F)F)CC1CC1)C(C)C c1(C(C(=O)NC(c2ccccc2)C)N(CCCF)CC)ccc(OC)c(OC)c1 c1(CN2C(C(N(CCO)CC)=O)C3CCC2C3)ccc2c(c1C)OCCO2 C1(NC(C(CN(C)C)(F)F)=O)CN(C(=O)C(=O)Nc2ncc[nH]2)C(C)(C)C1 c1(C(=O)NC(CNC(C(C)OCC)=O)CC)cc2sc(Br)cc2s1 C(CC(=O)NCC1CCN1C(N1CC(C(=O)NCC)C1)=O)OCC#C c1(OCC=C)ccc(Cl)c(C(=O)NCC2CN(C(c3cnsc3)=O)C(C)(C)C2)n1 C(CC(=O)NCCN(C(c1cnnn1C1CC1)=O)CC)(C1=CCCC1)OCC c1(COC)cccc(CC(N2CC3C(N(C(=O)C=CC4CCCC4)C)C3C2)=O)c1 N1(C(C2CCCC(C)O2)=O)CCC(C(=O)N(C)C)CC1(C)C N1(C(C2C(CC)C2)=O)CC2(CCC2CNC(C2(c3ccccc3)CCCC2)=O)C1 N1(CC(=O)N(C2CCN(C(C3CCN(CC)C3)=O)C2)C)CCN(C)C(=O)C1 C#Cc1ccc(C(=O)NC(C)CNC(c2sccc2C(C)=O)=O)nc1 c1(C(N2C(CNC(c3c(Cl)cc(C)nc3)=O)C=CC2)=O)cccc2c1C(=O)NC2 C1(COC)(NC(=O)C(=O)NC2CC2)CCN(c2ccnc(C)n2)C1 C(N=C(NCc1cc(Cl)cc(Cl)c1)N1CCC(SC)C1)c1cnn(CC)n1 C1(NC(C(CCC)CC)=O)CC2CCC(C1)N2C(=O)C(F)CCC(C)C C1(C(=O)NC(CNC(C2CC3CC2C3)=O)C2CC2)(OCC)CCCC1 C1(C#N)(CC(=O)NC(CNC(c2c(CC)csc2)=O)CO)CCCCC1 C(=O)(C1OCCc2ccccc21)NCC1(O)CCN(C(CC(=O)OC)=O)CC1 C1(CC(=O)N(C2CCCC(NC(c3n[nH]c(C)c3Cl)=O)C2)C)CC(=O)NC(=O)C1 c1(N2CCCC(CNC(c3ccc(Cl)o3)=O)C2)nc(Cl)nc2ccc(Cl)nc12 CC1=C(C(=O)N2CC=CC2CNC(c2c[nH]nc2F)=O)Cc2ccccc2O1 N1(C(C(C)OCC(C)C)=O)CC2(CCC(NC(c3cc(=O)cc[nH]3)=O)CC2)C1 CC(CCOc1ccccc1)C(=O)NC1CC(NC(c2cnnn2C2CC2)=O)C1 c1(OC)ncnc(C(N2CC(O)(CCNC(c3cccc(O)c3Cl)=O)C2)=O)c1F S(=O)(=O)(c1ccc(NCCOC(F)(F)C(F)(F)F)c(C#N)c1)NCCCC(C)CO c1(SC)cc(C(=O)NCC(C)(O)CNC(=O)CC2CC(F)C2)n(C)n1 C1(NC(=O)NCCc2ccc(COC)cc2)CCCC1S(C)(=O)=O c1(C(C)C)ccc(N2CCC(C(C)NC(=O)C(C)CF)C2)nc1 C1(C(=O)NCC2CCCC2NC(C2C3CCCC23)=O)CC2C=CC1C2 CC1(C)C(CNC(c2[nH]ncc2C#N)=O)CCN1C(c1ncccc1Br)=O N1(C(CCCSC)=O)CCC2OCCN(C(C3CC4CC3CC4O)=O)C2C1 N1(C(CCOC(CC(C)C)C)=O)CCN(C(=O)Cn2cnc([N+](=O)[O-])c2)CC1C C(=O)(C1CCc2nccn21)NC(C1CN(C(C(C(C)C)NC(N)=O)=O)C1)C C(=O)(CCCCCSC)NCC1N(C(CCC(=O)NCCC)=O)CC1OC c1(C(NOCC(=O)NCC(C)O)=O)cc2cccnc2[nH]1 CC(CC(F)(F)F)C(=O)N1CCCCCCC1C(N1CCC(C)(C)C1C)=O N1(C(c2c(C)n(C)cc2)=O)CC2CC(C1)N(C(=O)C(O)Cc1ccccc1)C2 N1(C(C2(CC=C)CCCC2)=O)CC(NC(c2cccn2C2CC2)=O)CC(C)C1 c1(C(N2CCC(C)(NC(c3ccc(OCC)cc3)=O)C2)=O)coc(S(N)(=O)=O)c1 Cc1cc(C(=O)NC2(C)CN(C(=O)CCCc3cccs3)C2)c(N)c(F)c1 Cn1ccc(-c2cc(C(N3CCC(CNC(=O)CC4(C)CC4(Cl)Cl)C3)=O)no2)n1 C(C(C)(C(=O)NCCC1(C)CCOCC1)NC(=O)Cn1cccn1)SC CC1CCC(=CC(=O)NC(C2CCCN2C(=O)CCNS(C)(=O)=O)C)C1 C#CC1(C(=O)N(CCC(C)C)C2CC2)CCN(C(=O)CNc2ccccn2)C1 c1(C(=O)NC2CC(CNC(C(C3CCOC3)SC)=O)C2)ccc(CC(C)C)cc1 N1(C(C2C(C)(C)C2NC(c2ccc(CF)cc2)=O)=O)CCC2(CCC(O)C2)C1 N1(C(c2cnc(C(C)(F)F)s2)=O)CCN(C(c2ccc(F)cc2O)=O)CC1CF C1(NC(c2cc(COC)on2)=O)CCCC(C(=O)NC2CC2c2ccco2)CC1 C1(NC(C(=Cc2cnc[nH]2)C)=O)CCCC(NC(c2ccsc2C)=O)CC1 c1(CC(N2C(C)CC(CNC(c3cc(C)sc3N)=O)C2)=O)c(C)ncnc1C n1(CC(N2CC(C)(C(N3CC(C(F)(F)F)C(F)C3)=O)C2)=O)cc(S(N)(=O)=O)cn1 CCC(C)CCC(=O)NC(C)CNC(c1cccc(OC(F)F)c1)=O C(C)(C)(CC(=O)NC1CN(C2CCC2)C1)N(C(c1c(OC)csc1)=O)C C12(C(N(C(C(=O)OC)C)C)=O)CCCC1CCN2C(c1c[nH]c(C)cc1=O)=O C1(OC)CN(C(c2cnn(C3CC3(F)F)c2)=O)CC1NC(=O)CCC#N C12(CNC(CCNC(C)=O)=O)CC(CN1C(C1CC(O)CN1C(N)=O)=O)C2 c1(-c2nc(CC3CCN(C(CSc4nc(C)[nH]n4)=O)C3)on2)nccnc1C N1(C(CSCCOC)=O)CCC(C(=O)NCC2CCCN2C)(C(C)C)C1 C1(NC2(CC=C)CN(C(=O)Nc3cc(COC(C)(C)C)on3)C2)CCCCC1C n1(CC)cc(CN(CC(=O)OC(C)=O)C(C)C)c(C)n1 CC1CC(C(N2CC=CC2(C)C(=O)N(C)C)=O)CN(C(=O)CCCC(=O)N(C)C)C1 C(=O)(C#CC1CCCCC1)NC1CCN(C(CSCC(C)C)=O)C1C N#Cc1cccc(C2CC2C(=O)NCC(O)CNC(=O)Cn2cncn2)c1 C(CCCCCNC(=O)C(COC)NC(C)=O)NC(CCOCCC)=O C1(CC(=O)NCCCCNC(C(C)(C)c2cccs2)=O)CC(=O)NC(=O)C1 C(=O)(C1CCCc2cc(C#N)ccc21)NC1CC(NC(C(CC=C)(C)C)=O)C1 CC(CN(C)C)CCC(=O)N(CCCNC(c1ccnc(N(C)C)c1)=O)C C(C)(C(C(C)C)NC(c1cc(C(C)C)no1)=O)NC(C(F)=C(C)C)=O C(=O)(C(=O)CC(C)CC)N1C(C(=O)NC(c2ncccn2)C)(CC)CCC1 C(=O)(C1=COCC1)N1CC(O)(C(C(=O)NCC(C2CCC(=O)N2)C)F)C1 N1(C(C2(C)N(C(C)=O)CCC2)=O)CC(NC(=O)C2=NOCC2)CC(F)(F)C1 N1(C(C)=O)CC(C)(CNC(c2ccc(C)c(NS(C)(=O)=O)c2)=O)CC1(C)C c1(CC)cc(C(=O)NCC2CC2NC(c2c(C)cnn2C)=O)ccn1 C1(NC(c2[nH]cc(C)c2)=O)CC2CC1N(C(C1(N(C)C)CCCC1)=O)C2 Cc1csc(=NCC(=O)NC2CCC(NC(=O)CC3CCOC(CF)C3)CC2)[nH]1 c1(CNC(CCCOC(CC)=O)=O)ccc(OCC(F)(F)F)cc1 C(=O)(C1=CCCCO1)NC1CCN(C(CC2(OC)CC2)=O)C1c1ccccc1 c1(CCNC(C2(C)CN(c3ncc4[nH]ncc4n3)C2)=O)c[nH]c2ccccc12 C1(C(=O)NC(CCOCC)C)CC(C)N1C(c1cn(CCO)nn1)=O c1(C(=O)NC2(C(=O)NCC(C)OC)CCC2)nc(C)c(C)s1 C=CCC(CNC(=O)CC1(O)CCC1)C(=O)NCc1cncc(OC)c1 C1(C(N2CCC(C)C2CNC(=O)COC2(C)CCOCC2)=O)CCC2(CCC2)O1 CC#CCC(C(=O)Nc1ccc(C2CC2)nc1)NC(=O)CC(=O)NC1CC1 O=C1NCc2cc(CNC3CCN(S(=O)(=O)c4cn[nH]c4)CC3)ccc21 CCC(C)CCCC(=O)N(C)CC1CCCN1C(c1ccoc1C(C)C)=O c1(C(=O)OCC)n[nH]c(=NC2CC(NC(c3ccsc3C)=O)C2(C)C)s1 C(=O)(C(C)CC(C)(C)C)NC1CCC(N(C(c2c(C)csn2)=O)C)CC1 c1(NCCCCC(C)NC(=O)C(O)C(C)(C)C)nc2c(cc1C#N)CCCC2 CC1(C)CCc2nc(C(=O)NCC3(O)CN(C(=O)C(=O)NC4CC4)C3)ccc2C1 C(=O)(C(C)(F)C(=O)N1CC2CC2(NC(=O)CNC=O)C1)OC C(=O)(C(CCC1CCC1)NC(=O)CCN=[N+]=[N-])N1C(CN=[N+]=[N-])CCC1 Cc1cc(CC(N2CC3CC2CC3NC(=O)CC2(CO)CC2)=O)cc(C)c1 c1(C(N(CC(C)(C)CNC(=O)CCC2CCCO2)C)=O)ccc2nc(O)oc2c1 N1(C(c2cc3[nH]ccc3s2)=O)c2ccccc2CCC1CN1CCOCC1 c1(NC(=O)Nc2c(C)cc(C(C)C)cc2)ccc2c(c1)CC(F)C2 c1(C(=O)NCC(C)CNC(=O)C(N2CCNC2=O)C)ccc2c(c1)CC(C)O2 C1(NC(C(C2CCN(C(CCCN(C)C)=O)C2)F)=O)CCC(C)(O)CC1 N1(C(C(C)N(C(C)=O)C)=O)CCCc2n[nH]cc21 CCC(CCOC)C(=O)NNC(=O)C(=O)Oc1ccccc1C O=C1CCc2cc(C(=O)NCCCCNC(C34CCCC(C3)OC4)=O)cnc2N1 c1(C(N(CCNC(Cc2ccc(C)nc2)=O)C)=O)n[nH]c2ccc(F)cc12 C1(CC)CN(CCCC2CC2)CCC1C(F)(F)F.C1(c2cncs2)C(=O)N1 C1(Cc2n(C)ccn2)CCCN(C(CCc2ccccc2)C(=O)NCC(F)F)C1 C1(C)(C(=O)NCc2cc(C(N3CC(CC#C)OCC3)=O)sc2)CCCN(C)C1 C(C)(CCN1CCOCC1)(c1nnnn1C1CCCCC1)NC(CC=CC)C C12(COCC)CC(C(=O)NC3CCN(C(=O)C=CC4CCOC4)C3CC)(CO1)C2 c1(CC)ccc(C(C(=O)NCC2CCOC2)N(C)Cc2cnc(Cl)s2)c(OC)c1 CC(=NO)c1cc(C(=O)N(C(C)CCNC(=O)COC2CC=CC2)C)cnc1O C1(NC(C2(C)COC2)=O)CN(C(C2(OC)CCC2)=O)CC1(C)C.OC CCCCC(C)CC(=O)N1CCN(C(C2CCN(C3CC3)CC2)=O)CC1C(F)F C(C(F)(C(=O)NC1CC(C)(C(=O)OC)C1)C(C)C)NC(C(C=C)CC)=O N1(C(C2C(C(=O)OC)C2)=O)CCC(C2CCCN(C(=O)C3=CCCSC3)C2)CC1 C1(n2c(-c3nc(OC(C)C)ccc3Cl)nc(C(CC)O)n2)CC(C)(C)OC1(C)C N1(C(CCC=C)=O)CC2CC(NC(=O)CCOc3cccc(C)c3C)C1C2 C(=O)(C(CO)C(F)(F)F)N1CC(CC(C)N(C(=O)COCP(C)(C)=O)C2CC2)C1(C)C C(=O)(CC(F)(F)C(F)F)NC1C2CN(C(c3n(CC)nc(C)c3)=O)C1C2 CCC(O)C(F)(F)C(=O)NCCCCCNC(=O)C(C)ONC(=O)OC(C)(C)C c1(C(=O)NC(C2OCCN(C(c3cc(C(C)C)sn3)=O)C2)C)ccn(C)c(=O)c1 c1(C(N(CC(CN(C(C(CCC)O)=O)C)O)C)=O)n[nH]c2c(OC)cccc12 C(C1=CCN(C(c2cc(C)ccn2)=O)CC1)NC(C(C)NC(COC)=O)=O C1(CCNC(C2(CCSC)SCCCS2)=O)CN(C(=O)CNC(N)=O)CC(C)O1 C1(CNC(c2cc(C)ns2)=O)CN(C(C2CC2c2nc[nH]n2)=O)CC1(C)C C(CC(C)NC(=O)CNC(=O)OC)NC(COCCOC)=O C(N=c1cc(CC2(Br)CC2)nc[nH]1)C1(CNC(=O)C2CC2)CCC1 C1(CCN(C(CC2C(CC)C2)=O)C)CCCCN1C(=O)COC(C)C c1(OC)cnc(CNC(=NCC2CCC2)NCC2(C)CCCCO2)cn1 CC(O)C(F)(F)C(=O)NCCOC1CN(C(=O)C(N2C(=O)CCC2=O)C)C1 c1(C(N2CC(C)(C(=O)NC3(C)CCS(=O)(=O)C3)C2)=O)cc([N+](=O)[O-])cc2c1OCC2 C(=O)(N=c1ccn(CC2CC2)[nH]1)C1(C)N(C(c2n(CC)ncc2)=O)CC(O)C1 N1(C(C2N(C(C)C)C(=O)COC2)=O)CC2C3CCC(C2C1)N(C(=O)C1CC1)C3 C1(CNC(C(=O)OCC)CCCF)CCC2COCCC2C1 O=C(CC1COc2ccccc21)NC1CCC(F)(CNC(=O)C(F)F)C1 N#Cc1c(NC(C2CCC(NC(c3ccnc4c3OCO4)=O)C2)=O)cccc1Cl c1(C(=O)NCCCCCN(C)C(c2cccc[n+]2[O-])=O)cncc(N(C)C)n1 CC1CCN(C(=O)C(N2CCOCC2CNC(=O)CC2CCCS2(=O)=O)=O)CC1 CC1CC(C)(C(N2C3CCC2CC(NC(=O)CCOC2CCC2)C3)=O)CC(C)O1 CC(CNC(c1cncc(Cl)c1)=O)C(F)C(=O)NCCc1cc(O)ncn1 c1(C(C)C)nc(N(C)CC2CC2(F)F)cc(N2CCSC(c3ccccc3)C2)n1 c1(C(=O)NCCC2CCCN(C(c3cc(CC)oc3C)=O)C2)ccc(F)c(O)c1 C(C(CS(=O)(=O)NCC(N1CCCCCC1)C)OC)OC N1(C(CCc2ncc(C)[nH]2)=O)CCC2CN(C(=O)C=CS(C)=O)CC2C1 C1(C(=O)NCC2N(C(c3ccnc(C)c3N)=O)CC2)CCc2ccccc2O1 N(C(=NCCF)N1CCC2C(F)(F)C2(C)C1)C1CCC(CCC)CC1 CC1CCCN(C(=O)C(=O)NC2CCCC(CNC(=O)CC3(O)CCC3)C2)C1 c1(C(=O)NC(CNC(CSCC#C)=O)CC)c[nH]c2ncnc(O)c12 C1(N(C(=O)C=C(Cl)Cl)C)CN(C(=O)Cc2cccc(Cl)c2)CCC1O c12cccc(c1)NC2=O.CCC(O)C(=O)NC1(C)CCOC1.C(=O)(C1CC1)N C1(OCCC(=O)NCC(CNC(CCNC(=O)OC)=O)O)CCCOC1 C1(CC=C)CCCCC1NC(C1CC(NC(C2(COC)CCC2)=O)CCO1)=O CC1CCN(C(=O)C(C)(F)F)CCN1C(C1CC(N=[N+]=[N-])C1)=O CCC(C)(C)C(O)C(=O)N1C(C(N2CCOCC2C(N)=O)=O)C2CC(O)C1C2 c1(OC)cc(NC(=O)CC2CC(NC(c3cc(C(C)C)on3)=O)C2)c(C)cc1Br c1(C(=O)NC2CN(C(C(CC=CCC)C)=O)C2)ccc(C(C)C)cc1C(C)C c1(C(N2CCN(C(c3c(CC)ncnc3)=O)CC2CC)=O)ccc2ocnc2c1 C(=O)(C(C)S(=O)(=O)C(C)C)N1CC(CNC(C(C)=C2CC2)=O)C(C)(C)C1 N1(C(c2c(C)n(C3CC3)cc2)=O)CCC(NC(c2ccoc2Cl)=O)C2(CCC2)C1 CC(C)CC(O)C(C)C(=O)NC1CC2(C1)CN(C(c1csc(CO)n1)=O)C2 N1(C(CC(C)c2ccco2)=O)CCN(C)C(CNC(c2cccnc2S)=O)C1 N1(C(C(CCNC(c2cc(O)cs2)=O)O)=O)CCC(F)(F)CC1 c1(N(CCC#C)CC2CCCC2CF)cccc(C(C)C)c1 C(=O)(CCC(CF)CF)N1C(C(=O)NC(CCN(C)C)(C)C)CC1 C(N=c1nc(N2CC=CCC(C)(C)C2)c2sccc2[nH]1)c1c(CC)nn(C)c1CC c1(NCC(C(C)C)N(C)C)ncc(S(=O)(=O)NCC2CC2)cc1Cl CC1CC(CNc2cccc(OC3CC3)c2)CN1c1nnnn1CCCCF CS(=O)CCC(O)C(=O)N(CC(CO)(CO)NC(=O)CC1(O)CCC1)C C(=O)(C(F)(F)CN(C)C)NCC1N(C(C(c2ccccc2Cl)C)=O)CC1 N1(C(C=CCC)=O)CC2CC(NC(c3oc(Br)cc3C)=O)CC2C1 c1(CC(=O)NC)noc(CCCl)n1.c1(CCNC2c3nnnn32)cc(C)on1 c1(C(C)(C)C)n[nH]cc1C(c1nnnn1C1CCC1)NCC(C)(C)C1CCCC1 Cc1nn(C)c(Cl)c1CC(=O)NC1CN(C(=O)CCOCC2CCCO2)CC1O Cc1cc(C(N2CCC(C3CCCN3C(C3CC(O)C3)=O)CC2)=O)n(C)n1 c1(C(N2C(C(C)C)C(NC(C3CCOC3)=O)CC2)=O)coc2cc(F)ccc12 C1(N2CCCN(CC(C)O)CC2)CCN(C(=O)OC(C)(C)C)CC12CC2 C(CO)(C(=O)NC(C1CCN(c2nnc(C(F)(F)F)s2)C1)(C)C)NC(C(C)C)=O c1(C(=O)NCCCCC(C)NC(=O)C(C)n2cccn2)ccc([N+](=O)[O-])cn1 [N-]=[N+]=NCCCCNC(C1C2CC2CN1C(=O)CN1CCC(F)CC1)=O c1(NCC(C(C)(C)C)OC)ncccc1S(=O)(=O)NCCCSCC(C)C c1(CN(c2ncnc3c(Br)csc23)C2C(C#N)CNC2)cccc(Br)c1[N+](=O)[O-] CCC(CC(=O)N1CC(CF)(NC(=O)CN2CC(=O)NC2=O)C1)SC c1(C(=O)NCCC2N(C(c3nc(C)n(C)n3)=O)CCC2)cc(F)c2[nH]nnc2c1 C(C1=NOC2CN(C(=O)CC(=O)N(CC)Cc3ncc[nH]3)CC12)NC(COC)=O N1(C(CC(C)(F)F)=O)CCCCC(CNC(=O)C=C(C2CC2)C2CC2)C1 c1(C(=O)NC2CCCC(N(C)C(c3cnsn3)=O)C2)nnc(O)c(Br)c1O C(C(O)C(=O)NC1CCC(CCC(=O)NCc2ncsc2C)C1)OC c1(NC(C2N(C(c3[nH]cc(C)c3)=O)CCSC2)=O)ccc([N+](=O)[O-])c(C)c1 Cc1n[nH]cc1CC(=O)NCC(C)(C)OCC(=O)N(C1(C)CC1)C N#Cc1cc(CN2CCOCC(C(=O)NCC(N3CCCC3)=O)C2)cc(Cl)c1 CN=c1nc(N(CC(F)(F)Cl)C)[nH]c(=NCCCc2nc3c([nH]2)CCCC3)[nH]1 N1(C(C(c2ccc(CC(C)C)cc2)C)=O)CCC2C(C1)CN2C(=O)CSC(C)C c1(CNC(=O)OC(C)(C)C)c(F)cc(Cl)cc1Br.Cn1ccc(=O)c(C=O)c1 N1(C(C(CSC)O)=O)CCC2(CC1)CC(NC(=O)C(C)OCc1ccccc1)C2 C(C(C)(C)C#CC(=O)NCC(C1CC1)N(C)C)NC(CC(C)C(F)F)=O c1(OC)ccc(C(O)C(C)NC(=O)CSc2cc(C3CCC3)ccn2)cc1 CC(C)S(=O)(=O)CC(=O)N1CCCC(C2(CNC(=O)CCCF)CCOCC2)C1 c1(C(C)N(CC#CCO)Cc2ccccc2)cc(F)ccc1OCCO N1(C(COC2(C)CCOCC2)=O)CCC2(CCCCC2NC(=O)CSC2CC2)C1 Cc1cc(Br)oc1C(N1CCC(CCNC(=O)CN2CCC(O)CC2)C1)=O N1(C(C(C)NC(N)=O)=O)CC(C(F)(F)F)C(CNC(=O)Cc2cnc[nH]2)C1 c1(C(=O)NCC2C(NC(c3ncn(C)c3)=O)CCC2)c(F)ccc(O)c1F c1(C(=O)NCC(C)(C)NC(CC2C(C)=NNC2=O)=O)c(O)nc(=O)n2c1CCC2 C(F)(C(F)(F)F)(C(F)(F)F)c1ccc(-c2nc(CC(C(C)(C)O)(C)C)on2)cc1 CC1CCc2onc(C(N3CCCC3C(C)NC(=O)Cc3cccs3)=O)c2C1 C1(NC(c2csc(-c3ccoc3)n2)=O)CCN(C(=O)C(F)CC2CC2)CC1F N1(C(C2CC=CC(NC(c3n(C)ccc3)=O)C2)=O)CCCCC(C)(F)C1 n1(CC(N2CC(OC)C(NC(=O)CN(C)C(C)=O)C2)=O)cnc2ccc(C)cc12 CCCC(CNC(C1CCCCC1(F)F)=O)C(=O)N1CCC2CC12C N1(C(c2ccc(CO)cc2)C(=O)NC)CCC(S(=O)(=O)c2ccc(Cl)cc2)CC1 c1(C(=O)NC2CCCN(C(c3c(CC)nco3)=O)C2)ccc2c(c1)C(=O)CCN2 CCN=C(NCCCc1nncn1C)NCC(c1cccc(F)c1)(C)C C12(CC(=O)NC(CCNC(CC(=O)NCC#C)=O)C)CCC(CC1)CC2 C1(NC(C2C(C)C2)=O)CN(C(c2ncc(Br)cc2Cl)=O)CC12CC2 CC(C)C(F)(CNC(=O)C1=NNC(=O)C1)C(=O)N1CCC(O)C(C)(C)C1 C1(C(=O)NC(CC)CNC(=O)CC2CCOCC2OC)CCC(=O)CC1C c1(C(=O)NCC(CNC(C(c2ccc(Cl)cc2)OC)=O)F)cn2c(n1)CCCC2 C1(CNC(CS(CC)=O)=O)CN(C(=O)CC2(c3ccon3)CC2)CC(C)(C)O1 c1(C(N2C(C)(CNC(CSCC)=O)CC(F)(F)C2)=O)ccc2c(c1)C(=O)NC2=O n1(CCC(=O)N(C)CC2CCN(C(CC(C)C3CCCC3)=O)C2)cnccc1=O c1(C(N(CC(C)(C)NC(C2CC3(CC(C)C3)C2)=O)C)=O)ccnc2ccsc12 CCCC(C)C(=O)NCCC(C)(C)CNC(=O)C(C)CCOC C1(NC(=O)C(CO)c2ccccc2)CCN(C(c2cnc(Cl)s2)=O)CC1 C1(C(=O)OC)(C(=O)Nc2cccc(-c3nc(C)cs3)c2)CC2(CCC2)C1 N1(C(=O)NC(c2cnc(C)s2)C)CCCC(N(C)C(=O)OC(C)(C)C)C1 C(CCCCCC(=O)NC1(c2ncccn2)CC1)NC(c1c(C)n(C)cc1)=O C1(F)(CNC(=O)OC(C)(C)C)CC(NC(=O)NCC2CC3(CC3)C2)C1 C1(NC(CC2(OCC)CCC2)=O)CCC(C(=O)NC(c2ncc[nH]2)CO)C1 C(CC(C)C(=O)N1CCC(Nc2ncc(OCCN(C)C)cn2)C1)=CCC N1(C(C2C(C(=O)OC)C2)=O)CCCC1C(C)(C)CNC(c1conc1C)=O N1(C(C(CCC)O)=O)CCN(C(=O)C(C)SCc2ccccc2)CC1C Cc1cc(C(N2CCCOC(CNC(=O)C3=CCOC3)C2)=O)c(C)n1NC(N)=O c1(CC(=O)NC(C2CCCN(C(C3(Cl)CC3)=O)C2)C)ccc2nonc2c1 C12(NC(C(C)CN(C)C)=O)CCCC1CN(C(=O)CCC(=O)N(C)C)C2 C1(OC)(CNC(=O)CC2CC3(CC3)C2)CCN(C(=O)C=CC(N2CCCC2)=O)C1 C(=O)(CCCF)N(CCNC(=O)CC1(O)CC1)CC CC1(C)CC(NC(c2csc(CO)n2)=O)CN1C(C1(C2CCC2)CC1)=O CCCCS(=O)(=O)N1C2CN(C(c3ccccc3C)=O)CC12 c1(-c2cn(CC3(CC)CCCC3)nn2)nnc2n1CCC2.N12CC(C(C)C1)C2 N1(C(C(C(C)C)C)=O)CCC2(CC(NC(c3c[nH]cc(Cl)c3=O)=O)C2)C1 Cc1ncc2n1CCN(C(c1cc(CNC(C3(C)CCC4CC4C3)=O)on1)=O)C2 c1(C(=O)NC2(C)CN(C(CCC=C(C)C)=O)C2)cnn(CC(C)C)c1C c1(CNC(C(c2c(C)nn(C)c2C)C)=O)cnn2c1CN(C(=O)CC(C)C)CC2 N1(C(C=CCCC)=O)CC(C2CCN(C(=O)CCN3CCCS3(=O)=O)C2)C1 N1(C(CSCC#C)=O)CC2(NC(=O)CSC)CC1C2 Cc1nc(O)nc(C)c1C(=O)NCC1CCCCC1NC(=O)C(=O)N1CCC1 C12(CNC(c3c(COC)cccn3)=O)CCCCC1CN(C(=O)C(C)=C(C)C)C2 C1(C(=O)NN(C)C)CCCN(CC)C1Cc1n[nH]c(-c2ccccc2)n1 N1(C(C2CCC(CNC(c3cnccc3CO)=O)CC2)=O)CCN2CCC1C2 c1(SC2(C(=O)NC(CNC(C(C=C)O)=O)C)CCC2)cc(C#N)c(SC)nc1C CS(=O)(=O)c1ccc(CN2CCC(n3cc(C4CCCC(F)(F)C4)nn3)CC2)o1 C1(CN(C(=O)C(CO)NC(N)=O)C)COCCN1C(c1ccc[nH]1)=O n1(C(CNC(C(C2CCN(C(C)=O)C2)C)=O)C)nc(C)cc1C N1(C(C(C=C)CC)=O)CCC(C=CC(=O)N(C)CC2(O)CCC2)CC1 N1(C(C2CCCN2CCC(F)(F)F)=O)CCC2(CC1)COC(CO)C2 c1(CCC)nc(C)c(C(=O)N(C2CCN(CC3C(C(=O)OC)C3)C2)CCC)o1 N1(C(C2(CCCC)CCC2)=O)CC(N(C(=O)CN(C)C(=O)OC)C)C(F)C1 N1(C(Cn2c(C)c(Cl)cn2)=O)CC2CC(Nc3ccc([N+](=O)[O-])cn3)CC1C2 c1(NC(CC2CCN(c3nccc(C)n3)CC2)=O)cc(Cl)cc(Cl)c1O c1(-c2nc(CC(CC)C)nn2CC(C)(C)CO)cnc2cnn(C)c2c1 C1(SC)CCC(N=c2nc3cnn(C)c3c(NCCN3CCCC3)[nH]2)C1 N1(C(c2ccc(C)cc2C)C(=O)NC)CC(n2ccnc2)C(C2CC2)C1 CC(C)(C)CCC(F)C(=O)N1CC(NC(C2C=CCS2)=O)C(O)C1 C(=O)(CCCC(=O)NCC(C)(C(C)C)NC(=O)Cc1cnccn1)N(CC)CC N1(C(=O)Nc2cn(CC=C)nc2)CCS(=N)(=O)C(C)C1 Cc1sc(O)nc1C(=O)NCC(C)(O)CNC(=O)C=C1CCC1 Cc1ccc(C(=O)NCCCCCNC(=O)CCOc2ccccc2)cc1 C(=O)(C(=O)NOC1CCC1)NC(CCC)C1CCCO1 CCC(C)CC(=O)C(=O)N1CCC(C2CC2)C1CNC(c1cnc2n1CCC2)=O CCCCC(CNC(C1(NC(C)=O)CCC1)=O)NC(C1CCN(C)C1=O)=O Cc1c(C(N2CC(NC(c3cc(F)c[nH]3)=O)C(C)C2)=O)ccc(F)c1[N+](=O)[O-] CC1(C)CCN(C(=O)C(=O)NCC(F)(F)F)C1CNC(=O)CC1CCCSC1 CC1(C)CN(C(=O)COCC(F)F)CC1CN=c1[nH]nc(C2CC2)s1 c1(NC(C23C(CN(C(Cc4cc(CC)no4)=O)C2)C3)=O)c(C)nc(C)nc1C C1(C(=O)NCC2N(C(c3cnc(CC(C)(C)C)s3)=O)CCC2)CCOC(=O)CC1 N1(C(C2C(C(C)C)CCO2)=O)CC2CCC(C1)C(NC(=O)COCC1CCC1)C2 N1(c2n(CCCOCC)c(COCC)nn2)CCC(S(=O)(=O)N2CCCC2)C1 c1(COC)ncc(C(=O)NC2CN(C(=O)CCP(C)(C)=O)CC2SC)c(O)n1 C12(C(N(CCCNC(=O)CSC3CCOC3=O)C3CC3)=O)CCCCC1C2(F)F n1(CC(N2CCC(C(C(=O)NCC3(COC)CCC3)(C)C)C2)=O)c(C)ccc1C CN1CC(=O)N(CC(N2CC3CC3(CNC(c3ccc(Cl)s3)=O)C2)=O)C1=O C1(F)(CNC(COCCC(C)C)=O)CN(C(c2cc(Cl)no2)=O)C1 c1(NC(c2ccc(NC(C3C(C(=O)OC)C3)=O)cc2)=O)ncc(OC)cc1Br C(=O)(CCCNC(N)=O)N(C1CCN(C(=O)C(O)Cc2ccccc2)C1)C c1(C(N2CC(NC(c3c(C)nc(CCC)o3)=O)C2)=O)cnc2c(F)cccc2c1 C1(C(=O)NCc2c(C(N(CC(=O)NC)C)=O)nco2)CC2CCC2C1 C(=O)(C(CC(C)C)NC(C1CCC(F)(F)C1)=O)NCc1ccc(C)s1 c1(COC)cc(CC(=O)NC(C)(C)CNC(=O)CN2CCC2C)no1 CCCC(C(=O)NC(Cc1ccco1)C(=O)N(C)Cc1nccs1)N(C)C N1(C(Cc2cnn(C)n2)=O)CC2(CCN(C(=O)CCc3ccc(F)nc3)CC2)C1 c1(C(=O)NC(C2CCN(C(=O)CCCC3CC3)CC2)C)c[nH]c2c(Cl)cccc12 C(=O)(CC(O)CN(C)C)NC(C1(O)CN(C(c2c(SC)csc2)=O)C1)C N1(C(c2[nH]cc(CC)c2)=O)CCCCC1CCNC(c1cc(C(C)(C)C)c[nH]1)=O C(=O)(CC(C)CC(=O)OC)NC1CN(C(C(CCC)=CCC)=O)CC1C(F)F c1(C(=O)NC(C2CCCCC2)C(=O)Nc2cn(CC#C)nc2)c(C)coc1CC C1(NC(c2ccccc2C(F)F)=O)(CO)CCCN(Cc2ccnc(O)c2)C1 C1(CC(N2CC(O)(CNC(C(C=C)c3ccccc3)=O)C2)=O)CCC(F)(F)CO1 CC(c1cccc(Cl)c1)=CC(=O)N(C1CN(C(=O)CC2OCCOC2(C)C)C1)C C(=O)(C(C(C)CC)c1ccccc1)N(CCNC(c1cc(C)sc1C#N)=O)CC C(=O)(C(CCCOC)NC(=O)C(CC)CCC)NC1(CC=C)CCCC1 C1(NC2CCC(N(C)C)C2)CCC2CNCCN2C1 c1(CN2C(CN3CCC(F)(C(=O)OCC)CC3)COCC2)cnc2ccccn12 c1(C(=O)NCC2(F)CC(NC(c3c(N)nc(Cl)cc3)=O)C2)cccc2sccc12 c1(OC)ccc2c(c1)OCC(C(=O)N1CC(NC(=O)CC3CCCCN3C)C1)=C2 c1(NC2CCC(C)CC2)cccc(C(=O)NC(CCOC)C)c1[N+](=O)[O-] c1(N(C)CC2CCCN2C(=O)C(c2ccccc2)F)nc2cc(Cl)ccc2s1 c1(N2CC=C(C)CC2)nc(N2CCN(C(C)(C)C)CC23CC3)c2[nH]ccc2n1 N1(C(c2c(C)ccs2)=O)CCC(C(C)(C)C)(CNC(c2snnc2C2CC2)=O)C1 c1(C(=O)NCCC2CN(C(C=C(CC)CC)=O)C2)c[nH]c2cc(C#N)ccc12 c1(N2CC(C#N)C(NC(c3ccc(C(F)F)cc3)=O)C2)ncnc2cnccc12 Cc1c(F)ccc(O)c1C(=O)N(C)CC1CCN(C(=O)CC2CC(C)(C)CO2)C1 N1(C(CCn2cc(CCCCC)nn2)=O)CCN(CC(=O)NCC(C)C)CC1 C1(C(=O)NCCN(C(C(C)S(C)(=O)=O)=O)C)CC2(C1)CC(F)(F)C2 C1(NC(C2C=CCCC2)=O)CCC2(CCN(C(c3ccn4cncc4c3)=O)C2)C1 C(=O)(C1=NOC(C)C1)NCCC1(NC(c2ccnc(C)n2)=O)CCC1 N1(Cc2onc(CCCC)n2)CC2CCC1CN2C(=O)C(C)c1cccs1 C1(O)(CC(N2CCCC(NC(c3cccc(C)n3)=O)C2)=O)COC(C)(C)C1 CN1CCCCC1C(=O)NCCN(C(C1CC(C)(C(C)(C)C)C1)=O)C1CC1 N1(C(=O)CC2CC2)CCCC(C(N2CCC(F)C2)=O)C1 C1(OCC(=O)NCCN(C(=O)CC2(O)CCOCC2)CCOC)CCC(C)CC1 C(c1ccc2[nH]ccc2c1)=CC(=O)NCCC1CCCN(C(C2C(C)(Br)C2)=O)C1 C1(C(N2CC(C)(CC=C)C2)=O)CC2CC2N1C(=O)C(O)C1CCCC1 c1(OC)nc(C)ccc1C(N1CC(NC(=O)Cn2ccc(=N)[nH]2)C(C)(C)C1)=O c1(SCCN2CCCC(C(N3CCCC3CO)=O)CC2)ccc2ccccc2n1 CN1CCCC12CN(C(C1CCCC1NC(=O)Cn1cccnc1=O)=O)C2 C1(C(=O)NCCC2CCCN(C(c3cnc(C4CC4)[nH]3)=O)C2)CC2CC(=O)C1O2 N1(C(C(C2CN(C(=O)C=CC(C)(C)C)C2)OC)=O)CCC(C2=NOCC2)C1 Cc1cc(C(=O)Nc2cnn(C3CN(Cc4ccc(C)nc4)C3)c2)cc(F)c1 C1(C(=O)NCCCCCCN(C(C(C(C)O)(F)F)=O)C)CCOC2(CCCC2)C1 Cc1cc(C)c2c(c1)N(C(c1nnn(C)c1C)=O)CCC2 C1(CNC(=O)COC(F)(F)F)CN(C(C2CCCS2)=O)CCC12CCOCC2 c1(C(C)=O)c(C)[nH]c(C(N2CCC(CNC(=O)C3CC3)C2(C)C)=O)c1C(C)C n1(C(C)C)c(O)nc(C(=O)NC(C(=O)NC(C)CNC(=O)C(C)C)CO)cc1=O N(C(=NCC1CC(C)(C)C1)NCc1ccco1)C(C1(O)CCCOC1)C N1(C(COc2cccc(OC)c2)=O)CCC(CNC(=O)C=C2CCC2)C(C)C1 c1(C(=O)NCCC2CC(NC(C3C(OCC)C3)=O)C2)cccc(C(C)(F)F)c1 c1(CNc2ccc(C(=O)NC3CCS(=O)(=O)C3)nc2)ccc(O)c(Br)c1 N1(C(CN2CC(=O)NC2=O)=O)CCCC2CN(C(C3(C(F)F)CC3)=O)CCC12 C1(CNC(C(CC)Oc2ccccc2C)=O)(CO)CCS(=O)(=O)CC1 Cc1ncc(C(=O)NCC(O)CNC(=O)CCc2nccn2C)cn1 c1(C(=O)NCC2(CC)OCCO2)cccn2nnnc12 n1(CC(=O)NCCCN(C(C2CCCC(O)C2)=O)CC)ncn2nccc2c1=O c1(C(N2CCC(O)C2COC)C(=O)NCCC)ccc(Br)c(Cl)c1 c1(C(=O)NC2(C)CN(C(C34CC=CCN3CCC4)=O)C2)cnn2c1C(=O)NCC2 c1(C(=O)NC(CN(C(c2cnc(O)n2C)=O)CC)C)cc(C)c2n[nH]cc2c1 C(N=c1[nH]c(Cl)nc2cc(C)sc12)C1CC(NC(C(CCCC)C)=O)C1 CCC(C)C(C)C(=O)NC(C)CN(C(=O)C(F)C(C)C)CC Cc1ccc(F)c(C(N2CC3CN(C(=O)Cc4ccnn4C)CC3C2)=O)c1O c1(C(=O)OC)ccc(CC(=O)N(CCCNC(=O)CC2CCCC(C)C2)C)cc1 CCC(C#N)(CC)C(=O)N1CCN(C(C2CC2Br)=O)C(C)C1 Cn1nc(I)cc1-c1noc(C2CC(C(F)(F)C(F)(F)F)C2)n1 N1(C(Cn2ccc(C)n2)=O)CC2(C1)C(NC(=O)C=Cc1ccsc1)CCS2(=O)=O c1(CC)ccc([N+](=O)[O-])cc1C(=O)NC1CCCCCC1NC(=O)CCC(N)=O c1(CCN(C(c2n(CC#C)ccn2)C(=O)OCC)C)ccc(C)cc1 c1(CNC(C2C(NC(c3cc(CCC)on3)=O)COC2)=O)ccccc1[N+](=O)[O-] N1(C(c2cc(C)ncc2)=O)CC(C)(C)OCC1CNC(=O)COCP(C)(C)=O C(C)(CCC(=O)N1CCCC1CSC)N(C(=O)Cc1c[nH]nc1C)C1CC1 CC(C(=O)NCC1C(CO)C1(C)C)C(C)NC(c1ccccn1)=O C(=O)(CC(F)(F)C(F)(F)F)NC(C(CO)NC(CCn1ncc(C)c1)=O)C N1(Cc2ccc(C)cc2)CCC2(CC1)CC2C#N.c12cn(nn1)C1(CC1)C(=O)NC2 C1(C(=O)NC2CCC(CN(C(=O)CC(F)(F)F)C)CC2)CC2CCC(C1)O2 CN=c1[nH]ccc(C(=O)NCC=CCNC(C2(F)CCOC2)=O)c1[N+](=O)[O-] C(=O)(CS(=O)(=O)CC1CCCO1)N1CC(OCCNC(C2(C)CCC(=O)N2)=O)C1 C(C1c2ccsc2CCN1C(=O)Cn1cccc1)NC(C(C=C)(C)CC)=O c1(C(=O)NCCCN(C)C(C2CCN2C(C)(C)C)=O)cc(-c2ccncc2)no1 C1(C)(C(=O)NCC2(C)C(NC(CCCC=C)=O)CCC2)CC(C2CC2)=NO1 S(=O)(=O)(CC(=O)NCCC1(OC)CN(C(=O)CC2CCS(=O)(=O)C2)C1)NC C12(NC(c3cnn(C(C)(C)C)c3Cl)C)CC1CN(Cc1cnccn1)C2 CC1CN(C(=O)CCn2ccccc2=O)CC(C)N(C(C2C3CCCC23)=O)C1 C(=O)(C1CCc2cc(Cl)ccc21)NC(CN(C(C1N(CC)CCC1)=O)C)(C)C c1(OC)cc(C(N2CCC(O)(C(C)NC(c3cc(C)[nH]n3)=O)C2)=O)cc(C)n1 C(C(F)(F)CCC(=O)NCC(C)S(C)=O)n1cc(CC(=O)OCC)nn1 c1(NCC(=C)Br)nc(N(C)Cc2ncc(Cl)n2C)nc2c1ncn2CC Cc1ccccc1CC(=O)NCCCOCCNC(C1(C#N)CCCO1)=O C1(F)(C(=O)NCC2C(C(=O)NC(c3cnc[nH]3)C)CCC2)CCOCC1 c1(C(=O)NCCC2CC(NC(c3ccc(Cl)s3)=O)C2)cnc(O)c2cncn12 c1(C(=O)NCC#CCNC(C(c2cccc(O)c2)C)=O)ccc2ccnn2c1 c1(C(=O)NCC2CCC(F)(CNC(CC(COC)C)=O)C2)ccc(Cl)nc1OC O=C(C1=CCN(C(C2(n3cccn3)CC2)=O)CC1)NCCCc1cncnc1 C1(CC=C)(NC(=O)CC2CC2(Cl)Cl)CCN(C(=O)C=Cc2ccncc2)C1 Cc1nccn1CC(=O)NCCCOCC(C)(C)NC(c1cnc(C2CC2)[nH]1)=O c1(OCC(=O)NC(CNC(c2cc(C3CC3)on2)=O)CO)ccccc1 c1(NC(C)=O)ccc(C(=O)NCC2CCN2C(=O)C(O)C(F)F)cc1Cl C1(N(C)C)CC(NC(=O)NCCCc2ncc[nH]2)C12CCC2 C(=O)(C1CCCc2ccccc21)N1CC(O)(CCNC(c2cnncc2O)=O)C1 C1(CN2CCC(N(c3nccs3)C)CC2)CC12CCCOC2 c1(C(=O)NC2C(F)CCN(C(c3c(COC)cc[nH]3)=O)C2)cccc(S(C)=O)c1 N1(C(CN(S(C)(=O)=O)C)=O)CCN(C(c2cnn3cnnc3c2)=O)C2CCCC12 c1(C(=O)NC(C(C)C)CNC(c2ccc(C3CC3)o2)=O)ccc(=O)n(CCO)c1 [N-]=[N+]=NC12CCC(C(=O)NC3(CO)CN(C(C4C=CCC4)=O)C3)(CC1)C2 CCC(CC)C(C)C(=O)N1CCC2CCCC12C(=O)NCCOC1CCOC1 C(N=c1[nH]c(=NCC2CC23CC3(F)F)[nH]c2cc[nH]c12)c1nc(O)cc(C)n1 C1(C(=O)NCc2cc(C(=O)NCCc3n(C)nnn3)no2)C2CC3C(C2=O)C13 Cc1cc(C)c(CC(N2CCCC(CNC(=O)CN(c3ccncc3)C)C2)=O)s1 Cc1ccc(CC(=O)NCC(O)CNC(C23CCC(CC2)CO3)=O)c(Cl)n1 N1(C(CCC)=O)CCCC2(CCN(C(C3CC4C(C3)C4(F)F)=O)C2)C1 N1(CC(CNC(c2ccc(OCOC)cc2)=O)O)CC(C)OC(C)C1 C(=O)(CC(F)(F)C(F)(F)F)N1CC(NC(C(C)C(=O)N2CCCC2)=O)C(F)CC1 c1(C(=O)NC2CC(C(=O)Nc3cnc(C(F)F)cn3)C2)cc(Cl)cc(Cl)c1Cl C(=O)(CC1=NN(C)C(=O)C1)N1C(C(=O)NC(c2ncc[nH]2)CC)CC1 c1(C(=O)NC2C(CNC(C3(C(C)C)CNC(=O)C3)=O)C2)cc2c(cc1O)OCO2 N1(C(c2c(C#N)ccs2)=O)CCN(C(c2cnn[nH]2)=O)CC(CO)C1 CN=c1nc(C(N2CC(F)(F)CC2CCNC(C2CC(F)C2)=O)=O)cc(C)[nH]1 N1(CCNC(C(=O)Nc2c(OC)ncnc2OC)=O)C(=O)NC(C)(C)C1=O C(=O)(CC(O)C1CCCC1)NC(C1(c2ccc(Cl)s2)CC1)C.C12CN(C1)C(=O)N2 C(=O)(CCC(=O)NN(C)C)NCC1C(CNC(c2ncc(C)cc2C)=O)C1 C(N=c1[nH]c(C)nc2c1CCCC2)C1(OC)CCOC1 C1(NC(CC2(N(C)C)CC2)=O)CCCC12CN(C(c1ccccn1)=O)C2 N1(C(=O)NCc2ccc(C(C)C)[nH]2)CCc2ncn(C)c2C1 C1(CNC(COC2CC(N(C)C)C2)=O)C=CCOC1.C12(CCC1)C(=O)N2 C1(C#N)(C(N(C(CC)CNC(C2CCCN2CC)=O)C)=O)CC12CCC2 c1(C(N2CC(N(C)C(c3ncccc3N)=O)C(C)(C)C2)=O)ccccc1S(C)=O N1(C(c2c(SC)ccs2)=O)CCCC2(CCC(NC(C3(CO)CC3)=O)C2)C1 c1(C(=O)NCC(CNC(COC(c2nccn2C)C)=O)CO)cnc2n1CCC2 c1(C(N2CCC3(CC2)CN(C(C2CC2F)=O)C3)=O)cc2ccc(Br)cc2cn1 N1(C(c2c(NCC)scn2)=O)CC2(CCN(C(=O)C(c3ccccc3F)F)C2)C1 C1(CNC(C2(OC)CCSCC2)=O)CC2(CO1)CN(C(=O)CCC1CC1(F)F)C2 O=S(=O)(c1cccnc1NCCc1cccs1)N1CCN(CCCF)CC1 CC(C)CC(C)(CNC(C1C2CCOCC12)=O)NC(=O)C=Cc1cnccn1 Cc1ccc2sc(N3CCCC(NC(=O)CCCC(N)=O)C3C)nc2c1 n1(CC)nc(C(=O)NC(C)CN(C)C(c2sc(C)cc2C)=O)cc1O C1(C(C)NC(C(C)NC(=O)NC)=O)CCCN1C(=O)CCCc1cccs1 N1(C(C2CC3CCC2C3)=O)CCN(C(c2cc(F)c(F)c(F)c2)=O)C2CCC12 N1(CC(N2C(CCNC(C3(C)CS(=O)(=O)C3)=O)CCCC2)=O)CCC(=O)NC1=O C(CCCCCNC(=O)C(c1cccc(Cl)c1)O)NC(C(C)OCOC)=O CCCC(C(=O)NC1CN(C(=O)C(C)(C)CO)CC1C)c1cccc(Cl)c1 C(CC(C(=O)N1CCC(CCCNC(c2cccc(C(N)=O)c2)=O)C1)OC)OC c1(C(N2C(CNC(c3c(COC)nc(C)[nH]3)=O)CC(O)C2)=O)ccc(Cl)cc1Cl N1(C(=O)CCCc2ccsc2)CCCC(CN(C(c2ccc(F)cn2)=O)C2CC2)C1 c1(C(=O)NCC(CO)NC(C(C)SCCCC)=O)cc(C(C)C)[nH]c1C(C)C C1(CNC(C(C)OC)=O)(NC(c2cc3c(s2)COCC3)=O)CCC(F)(F)CC1 N1(C(C2N(C(Cc3c(CC)con3)=O)C(C(C)C)CC2)=O)CCC2(CCCC2)C1 c1(C(=O)NC(CN(C)C(C2CCC2F)=O)(C)C)cnn(CCO)c1 Cc1nn2c(c1C(=O)NCC1CC(NC(=O)C(C)C3CCC3)C1)CCCC2C C(=O)(CCCC(C)(C)C#N)N1CC(OCC(C)NC(CCCCCOCC)=O)C1 C1(C(CNC(=O)CC=CC(C)(C)C)NC(CCN(C)CC)=O)CC=CCC1 C1(OC)CCC2CN(C(C(=O)NC3CC3)C3CCC3)CC12 C#Cc1cc(F)ccc1CN1CCCC(C)(C(=O)Nc2ncccc2O)C1 C(=O)(CC(C)CC(=O)N1CCCOC(CNC(=O)CCCn2cccn2)C1)OC C(=O)(CCCC(F)(F)F)Nc1scc(C)c1C#N.c12nc(cn1C)NC2=O c1(CNC(C(N2CCC(c3nc(C)on3)C2)C)=O)cn(C)nc1C1CC1 CCCC(CC(=O)N1CC=CCO1)NC(c1ccc(C)c(C#N)c1)=O c1(C(=O)NC2C(CNC(=O)C=C3CCOCC3)CC2)n[nH]c2c1CCC2 Cc1cc(N2CCCC2)ccc1C(N1CCC(NC(=O)C(C)(C)C#N)CC1)=O CC(C(=O)N1CCCC(C2CCN(C(=O)CC#N)CC2)C1C)S(N)(=O)=O c1(C(=O)NC2CN(C(=O)CCCCCF)C3(CCC3)C2)cc(F)cc2nn[nH]c12 CCC(C(=O)NC1(CCCNC(=O)C(O)Cc2cnn(C)c2)CC1)N(C)C Cc1ccc(CC(=O)NCC(O)CCNC(=O)C(C)c2cccs2)c(C)c1 C#Cc1ccc(C(N2C(C(N3CCC34CN(C)C4)=O)CC2C)=O)nc1 N1(C(CC(C=C)C)=O)CC23CCCCC2(C1)CN(C(c1nc(C(C)C)cs1)=O)C3 C1(C(C)C)CCC(C)CC1C(=O)OC(=O)C(C)Sc1cccc(Br)n1 c1(C(N2C(C(=O)Nc3c(C(N)=O)cc(I)cc3)CC2)=O)cccc2nscc12 CC1CCN(CCNC(=O)NCC2(CO)CCCC2O)CC1 N1(C(c2c(C(C)C)ocn2)=O)CC2CN(C(C3(C4CCCO4)CC3)=O)CC2C1 Cc1sc(C(=O)OC(c2ccc(OC(F)F)cc2)C)nc1C(F)(F)F S(=O)(=O)(c1ccc(Cl)c(C(=O)NCCCNC(=O)CC2(O)CCCCC2)c1)NC Cc1onc(CC(=O)NC2(CNC(C3(N(C)C)CC(F)(F)C3)=O)CC2)c1C#N N1(C(c2ccc(C#N)o2)=O)C2COCC1CC(NC(=O)CC1CCCSC1)C2 C12(CC(=O)NC3C=CC(CNC(C4CCCC45CCC5)=O)C3)CCC(CC1)CC2 c1(N(C)C)ncc(C(=O)NC(CNC(C2COC3(CCC3)C2)=O)CO)cc1Cl c1(CC(C)C)ccc(C(=O)NC2CCCC2NC(=O)CC(C)n2ccnc2)s1 c1(CC(=O)NCC2(F)CN(C(c3ccc(CC)[nH]3)=O)C2)ccc(CC)cc1F C#Cc1c[nH]nc1C(=O)NCC(C1CCCCC1)NC(C1(Cl)CC1(F)F)=O N1(C(C(CC#C)O)=O)CC(CC(=O)NCCCOC(F)(F)F)C2(CC2)C1 Cc1nnn(CC(N2CC(CC(C)NC(C3(C(F)F)CCCO3)=O)C2)=O)n1 C1(C(=O)NC2(C(C)(C)C)CC2)CC(NC(=O)CC2CC3C=CC2C3)C(O)C1 N1(C(COC(CC)CC)=O)CCCC(C)(CNC(C2CC(CC(C)(C)C)C2)=O)C1 C(=O)(C1(C)OCCc2ccccc21)NC(CC)CNC(c1nc(C)ccc1O)=O C=CCC(C)C(=O)N(C)CCC1CCN(C(=O)C(C)(C)COCCN(C)C)CC1 CCCCC(O)C(=O)NCCCOCCNC(=O)CC(C)Cc1cccc(F)c1 C1(C2CCN(C(c3ccccc3N(C)C)=O)C2)(NC(c2nnc(C)s2)=O)CC1 C1(NC(c2sc(C)c(O)n2)=O)C(C)CCN(C(c2csc(C)c2N)=O)C1C C12(C(=O)NCC(CNC(c3c(OC)scc3)=O)C)CCC(C1)OC2C N1(C(C=CSC)=O)CC2CC3CC2C1C3NC(C1CC2CCC(C1)C2O)=O C1(NC(CC2CC(N(C)C)C2)=O)C2CC1N(C(C13CC(F)C1C3)=O)C2 C1(NC(CCn2c(C)ncc2)=O)CCN(C(c2ccccc2F)=O)C1C C1(OC)CC(NC(c2cocc2C)=O)CN(C(C2CC=CCC2)=O)C1 C(=O)(C1COc2ccccc21)NC(C(C)C)CCNC(=O)CC1CC2CCC1O2 N1(C(C=C(CC)C)=O)CC2CCCC2(NC(=O)C(O)CC2CCCCC2)C1 N1(C(=O)NC2CC3COC2C3)CCCCCCCCCC1 c1(OC)cnc(Br)cc1NC(C1CC12CN(C(=O)CN1CCOCC1)C2)=O c1(C(N2CC(C)N(C(C3CCCC(C#N)C3)=O)CC2)=O)ccc2c(c1)CCO2 C1(C(=O)NCCN(C(c2cnn(CC(F)F)c2)=O)CC)CCC2(CC2)C1 c1(C2C(C(N(C3CCN(C(=O)CNC(c4ccsc4)=O)C3)C)=O)C2)ccccn1 c1(C(=O)NCC2(Nc3c(C)cnc(Cl)n3)CCCC2)ccc2[nH]ccc2c1 c1(C(=O)NCC2(O)CC(O)C2)coc2c1CN(C(C1(O)CCOC1)=O)C2 c1ccc(C)c(Br)c1C.c1(C(N2C(=O)CN2C=O)=O)ccc[nH]1.C1(C(=O)OC)CC1 C(CNC(=O)CCc1cccn1C)(C(=O)N1CCC1)N(C)C CC1CN(C(=O)CC(C(C)(C)C)NC(c2ccco2)=O)CC(C)(C)CO1 CCCC(C)CCCC(=O)N(C1CCN(C(=O)CCc2cc(OC)no2)C1)CC C1(NC(C2(C)CC=CCO2)=O)CN(C(=O)CN2C(=O)CCC2=O)CC1C1CC1 N1(C(c2nnn(C)c2N)=O)CCN(C(C2CS(=O)C2)=O)C(CC(F)F)C1 CC(C(=O)N1CCC(n2cc(CNC(=O)C3CC3)nn2)C1)C(F)(F)F Cc1c(Br)cc(C(C(=O)NCCC2CC2)N(C2C3COCC23)C)cc1[N+](=O)[O-] Cc1cccc2[nH]c(C(N3CCCC(NC(C4CC(N(C)C)C4)=O)CC3)=O)cc12 CCCCCCC(CC)C(=O)N(CC(C)NC(=O)CSc1cnn(C)c1)C C(=O)(C(C)(C)CCCNC(=O)CCCCC(C)C)NCC(C)OCC#C CCCCC(O)C(=O)N1CC2CC1CC2CNC(c1ccc(CC)cc1N)=O c1(CNC(C(N)Cc2cc[nH]n2)=O)nc2c(s1)CCCC2 CC1=NOC2(CCN(c3ncccc3S(=O)(=O)NCc3ccoc3C)CC2)C1 C1(C2CC2)(C(=O)NCc2ccc(C(=O)NCCP(C)(C)=O)o2)CC(=O)C1 Cc1cc(F)c(C(N2CC(C3CN(C(c4ccnnc4C)=O)C3)C2)=O)c(Br)c1 C=CCC(CC(=O)N(C)CC1CCCCC1)NC(C1(C)CCC2CC2C1)=O N1(c2c(CC)cnc(Cl)n2)CCC2(CC1)OCCCC2NC(c1cc(C)ns1)=O O=S(=O)(c1ccc(=NCc2ccc(C3=CCNCC3)cc2)[nH]c1)N(C1CC1)C1CC1 C#CCC(CC#C)C(=O)NCCOCCN(C(=O)C(C)n1cccc1)C c1(C(=O)NC(CCN(C(C(CC)c2cccnc2)=O)C)(C)C)cccc(Cl)c1 CC1CN(C(C2(NC(=O)CCc3cn(C)cn3)CC(F)(F)C2)=O)CC(C)S1 C#Cc1cccc(C(=O)NCC(C)(C)CNC(=O)CC2CCC(C)CC2)c1F c1(CC)nc(C)ncc1C(=O)NCCC1CCC(NC(=O)C2CC2)C1 N1(C(=O)NC(C(C)C)c2cccs2)CCC(Cc2ccoc2)CC1 c1(C(=O)OC(C)=O)ccc(C(=O)NCC2(c3cn(C)nn3)CC2)o1.C1CCOC1 CC1CN(C(=O)OC(C)(C)C)CCC1CNc1ccc(C2CN(C(N)=O)C2)nc1 CCC(C(=O)NC(COC)C(=O)NC(C)CF)C(C)(C)CC Cc1cc(O)ccc1CC(=O)NCC1(NC(=O)CCc2ccc[nH]2)CCCC1 Cc1nc(=N)[nH]cc1C(=O)NCC1COCC1NC(=O)CC1(O)CCCOC1 C(c1cnccn1)=CC(=O)NCCCCN(C(C(c1cncnc1)C)=O)C c1(C2(C)CC2)nc(C2CCCC2)nn1-c1ccnc(Cl)c1 C#Cc1cnc(C(N2CC3(CC3)CC2CNC(=O)Cc2ccsc2)=O)c(C)c1 c1(C(=O)NC(C(C(C)C)NC(CSCC)=O)C)c2c(nc3ccccc13)CCC2 CC1CN(C(c2ccc(Cl)cc2CO)=O)CC(C(N)=O)O1 O=C1CC2CC1NC2NC(c1ccc(C(F)(F)C(F)(F)F)cc1)=O C1(NC(Cc2ccc(CSCC)cc2)=O)CCCCN(C(=O)C(C)SC)C1 C1(C)(CC)C=C(C(=O)NCC(C)(CC(C)C)NC(c2ccc(C(N)=O)cc2)=O)C1 c1(C(N2CCC(N(C(CCCSC)=O)C)C(C)C2)=O)ccn2[nH]c(=N)nc2c1 CC(N=c1cc[nH]cc1)C(=O)NCC1(CNC(=O)COCC2CCC2)CC1 C(N=c1cc[nH]cc1C#N)C1OCCCN(C(C2CC(CC)(CC)C2)=O)C1 N1(CCC)CC(=O)N(CSC)C1=O.C1(OCCC)CCCCC1 C(CCN=c1[nH]c(=NCC2CCC(O)C2)[nH]c2ccc(Cl)cc12)NC(=O)NCC C12(OC)CCCC(C(=O)Nc3cnccc3C(c3ccc(F)cc3)=O)(CC1)C2 C1(C(N(CCCNC(c2ccoc2)=O)C(C)C)=O)CCC(=O)N1C1CC1 C#Cc1ccc(NC(=O)NC2CCCC2C)c(Br)c1 N1(c2c(C)cncn2)CC2CCC(NC(C3(C)CCCCCC3)=O)CC2C1 C(C(CC(F)(F)F)NC(=O)Cc1ccoc1C)NC(C1N(CC)C(=O)CC1)=O c1(Cn2c(-c3c(C=CC(=O)OC)cccc3)ncc2)cnc2ccccc2c1 C1(CNC(C2CCCN2c2ccccc2)=O)CCCN1C(=O)Cn1cnnn1 C1(NC(=O)CCC2CCOC2)CN(C(=O)CC2(O)CCC2)CCC1F c1(CC(C)C)cc(C(=O)NC2CC2NC(c2sccc2Br)=O)n[nH]1 C(=O)(CCCS(N)(=O)=O)N1CC2C(NC(c3cncc(SCC)n3)=O)C(C2)C1 C1(C(=O)NC(c2ccccc2)CC)CN(C(C)C2CC2)CCC1(F)F C1(CC(=O)NCC(C)CNC(c2cnsn2)=O)CCCC(O)C1 CCC(CC(=O)N1CC(CNC(c2cncs2)=O)CC1(C)C)C(F)F Cc1cccc(C(=O)NCC2(C)CCN(C(=O)C=CC3CCOC3)C2)c1C C(=O)(C#CC1CCOC1)NCCCCN(C)C(c1ccnn1C)=O C1(CCC(=O)NCCC(CNC(c2c(C)nco2)=O)O)CCCC(=O)N1 C1(C(=O)NCCC(CNC(=O)CC(C)(C)OC)OC)C2CCC(F)C12 CC(C)(C)CCC(=O)N1CCC1C(=O)NC1(C)CCN(C(=O)OC(C)(C)C)C1 C12(C(=O)NCC(C)NC(c3cc(O)nn3C)=O)CCC(C)(C(=O)O1)C2(C)C C(CCCCCNC(c1ccc(-c2ccc(C)nn2)cc1)=O)NC(C=NOC)=O N1(C(Cn2c(N)cc(C)n2)=O)CCC(C)C(CNC(c2cc(=O)n(C)cn2)=O)C1 n1(CC)cnc(C(C(=O)NC)N(C(COC(C)(C)C)C(=O)OC(C)(C)C)C)c1 C1(C(=O)NCCCN(CCCCNC(C2CS(=O)(=O)C2)=O)C)CC12CC(O)C2 C1(CC(=O)N(CC(O)CNC(=O)C=Cc2cnc[nH]2)C)CCC(C(N)=O)CC1 c1(N(CCCN(C(c2cc(SC)oc2)=O)C)C)nc2cc(C)ccc2o1 CC1(Cn2cc(CN3CCS(=O)CC3)nn2)CCCCNC1=O S(=O)(=O)(c1ccsc1C(=O)NCC(CO)NC(C1(C)CC1(C)C)=O)N(C)C c1(C(C)(C)C)ncc(C(=O)NCC2CCN2C(=O)COC2CC(F)(F)C2)o1 C(C(C)(C)CNC(=O)C(C)N(C(=O)C(n1ccc(C)n1)C)CC)OCC c1(NC(=O)Nc2ccco2)cc(NCC=CCN2CCOCC2)ncn1 N1(C(c2c(OC)nsc2)=O)CC(NC(=O)CC2COCCO2)CC(C)(C)C1 c1(C(=O)NCC)c(C)nsc1N.C(=O)(CC=CCNC(=O)NNCC)OC C1(C(=O)NCC2CCCOC2)CC(F)CN1C(c1n[nH]cc1Cl)=O Cc1cnc(NC2CCCC2CCO)c(S(=O)(=O)N2CCCC(C(C)C)C2)c1 C(=O)(C(C)S(=O)(=O)C(C)C)NC(C)CCNC(c1n[nH]c2c1CCCC2)=O C1(CC(=O)NC2C(NC(CC3CN(C)C3)=O)CCC2)CC(C)(C)OC1=O c1(CC(=O)NC(C)CCN(C(=O)C(C)CC2CCC2)C)c[nH]c2nccc(Cl)c12 C(=O)(C1=CCCCO1)N(C1CCC(NC(C2(CO)CCOCC2)=O)CC1)C C1(F)(C(=O)NCCCCCN(C(c2n(OC)cnc2C)=O)C)CC12CCCCC2 Cc1cc(C(=O)NCC2(NC(c3cccnc3O)=O)CC3CCC2C3)cc(F)c1 c1(C(=O)NCCN(CCOC)C(C2(C)C=CCCC2)=O)cc(Cl)cn1C C1(NC(C2CCCC(N)C2)=O)CN(CC(=O)Nc2ccccc2Cl)CCC1O N1(C(c2ccc(C#C)cc2)=O)CCC(CNC(=O)Cc2cnc[nH]2)C12CCC2 n1(CC(C)C)ncc(C(=O)N(CCc2ccc(Cl)s2)Cc2ccco2)c1C(F)F CC(C)(C)CCC(F)C(=O)N1CC(CNC(=O)COC2(C)CCC2)C2(CCC2)C1 C1(C(=O)NC(C)CN(C(=O)CN2CCN(C3CC3)C2=O)C)CCS(=O)(=O)C1(C)C c1(NC(C2N(C(C(C)(C)C)=O)CSC2)=O)cc(Cl)ncc1Br O=C(CCCCc1cnn[nH]1)N1CCN(C(C2(CC(F)F)CCC2)=O)CC1 N1(C(CCOCC#C)=O)CCSCC1C(N1CCC(F)(C(=O)OC)C1)=O N1(C(c2cc(OC)n[nH]2)=O)CCC(NC(=O)C(O)Cc2[nH]cnc2C)C1C C1(C(=O)NCC2(COC)CC2)CC(F)CN1C(c1ccon1)=O N1(C(CN(C(=O)C(C)Cc2cnn(C)c2)C(C)C)=O)CCc2sccc2C1 N1(C(C2CN(C(COC(C)C)=O)CC(C)(C)C2)=O)CCn2c(O)nnc2C1 CC1(C(=O)NCC#CCNC(c2ncoc2C(F)(F)F)=O)CCCC1 N1(c2snc(CCOC)n2)CC2(CN(C(C3CC(C)(F)C3)=O)CC(C)(C)O2)C1 C(=O)(CS(=O)C(F)(F)F)NC(C)CC1CN(C(c2cncc3c[nH]nc23)=O)C1 n1(CC)nnc(C)c1C(=O)N(C)CC1CCN(C(=O)C(C)Cc2ccco2)CC1 C1(CCN(C)C(C2C3COCC23)=O)CCN(C(c2cc(O)nn2C)=O)CC1 C1(COC)CN(C(c2ccc(C(C)(C)C)c(Cl)c2)=O)CCN1C(=O)C(C)O N(C1C(=O)N(C)c2ccc(Br)cc21)C(c1n(C(C)C)cc(Br)c1)=O CCC(C)C=CC(=O)NC(CN(C(=O)C(F)=C1CCC1)C)CC c1(C(=O)NC(C(C)C)CNC(c2cnn[nH]2)=O)ccccc1CC#N CCCC(C(=O)N1CCCC(N(C(=O)Cc2cccc(C(F)F)c2)C)C1)OCC c1(CC(=O)N(CCCCNC(Cc2scc(CC)n2)=O)C)c(C)cc(C)cc1C C1(NC(C(C)(C)C(N)=O)=O)CN(C(=O)C2=CCCOC2)CC2(CCC2)C1 C1(C(=O)NC(C2CN(C(C3CCC3C#N)=O)C2)C)(CC)CCOCC1 c1(C(=O)NCC2CC(NC(CCCCC#C)=O)C2)cc2ccccc2nc1OC C1(NC(CCCC(=C)C)=O)CC1C1CCCN(C(=O)CCC2CCCN2C)C1 C(=O)(C1=CN=C2N=CNN2C1)NC1(CNC(c2cnc(COC)s2)=O)CC1 c1(C(C)N(C(=O)C(=O)NC2CC(=O)N(CC(N)=O)C2)C)ccc(C2CC2N)cc1 Cc1nn2c(c1C(=O)NC1C=CCC1)OCCCC2 CCC(CC)C(F)C(=O)NCCOC1CN(C(c2ccccn2)=O)C1 N1(C(C2(NC(c3ccc(C)nc3O)=O)CC(F)C2)=O)CC(CO)CC(C)(C)C1 N1(C(CCC#CC)=O)CCN2CCN(C(=O)C(CC(C)C)NC(C)=O)CC2C1 C1(N(C(c2c(OC)cccn2)=O)C)CCN(C(=O)C(O)C2CCCC2)CC12CC2 CC(C)(C)C(O)C(=O)N1CCCC1C(C)(C)C(=O)N1CC(F)(C(N)=O)C1 N1(C(C2C3CCN(C(C4CN(OC)C(=O)C4)=O)CC32)=O)CC(C)C12CCOCC2 C(=O)(C(C)(C)C(C)(F)F)NCC(CNC(CCOC)=O)C(F)(F)F C(C(COC)C(=O)N(CCC(=O)NCC(O)CC(C)C)C(C)C)OC c1(C(N2C(C(=O)NC(c3ccc(Cl)cc3)C)COCC2)=O)ccc2c(c1)OCO2 C1(NC(=O)Cc2ccc(Cl)nc2)CN(C(c2cc(Cl)c[nH]2)=O)C2(CCCCC2)C1 c1(-c2n3c(nn2)C3)cc(F)c(F)c(F)c1.N1(CCCOC)CCC(CCF)CC1 c1(CC)cncc(C(=O)N(C2CC(NC(=O)CCOc3cccc(F)c3)C2)C)c1 Cc1cc(F)ncc1C(=O)NCC1C2CN(C(C3CCC(=O)C(C)C3)=O)CC12 C1(CNC2CCCCN(C(CSCC)=O)C2)CC12CCC(F)(F)CC2 C1(CNC(c2cnc(CC)s2)=O)CC(F)CN1C(c1cnn(C2CCC2)c1C)=O N1(C(C2N(S(C)(=O)=O)CCCC2)=O)CCCCC(CNC(=O)Cc2cnco2)C1 C=C(C)CC(C)C(=O)N1CCCOC(c2ccccc2Cl)C1 C1(OC(=O)NC)CN(NCCCC(C(C)(C)C)NC(=O)NC)C1 O=C(C1=CCC(F)(F)CC1)NCCC1(O)CN(C(c2cn3c(n2)CCCC3)=O)C1 Cn1ccc2ccc(C(N3CCC3CNC(c3cnc4[nH]ccc4n3)=O)=O)cc12 CC1CN(C(=O)C(C)(C)NS(C)(=O)=O)CCC1NC(=O)C(=O)C(C)(C)C C1(CC(C)C)(C(=O)NC2CCC2C(=O)N(CCCn2nccn2)CCO)CCC1 C1(CNC(CN2CCCC(CC)C2)=O)CN(C(=O)C#CC2CCC2)C(C)(C)C1 CC(O)(Cc1ccccc1)C(=O)NC1CCCCC1NC(c1cc(Cl)cs1)=O C(=O)(C(C)(C)CC(=O)NCC1CN(C(=O)COCc2cccc(Cl)c2)C1)OC c1(C(=O)NC2CN(C(C(COC)(C)OC)=O)CC2C)cnc(C)[nH]c1=N n1(CCC)nnnc1C(c1cncn1C(C)C)NC1CCCC1F C1(N(C(C(CC=CC)C)=O)C)CC2CCC(C1)N2C(c1ccc(COC)s1)=O c1(C(=O)NC(CC(C)NC(c2n[nH]c(=N)[nH]2)=O)C)ccc(-c2ccncc2)cc1 c1(CC(=O)NC2CC(NC(C(C)NC(CC)(C)C)=O)C2)ccc2c[nH]nc2c1 C(C(O)CCNC(c1cc(C)ns1)=O)NC(C(C)NC(=O)NC)=O CC(C)(C)CCC(C(=O)O)NC(c1cc(Cn2cc(C(O)C3CC3)nn2)on1)=O c1(C(=O)NCCCC(C)NC(C2CC(=O)C2)=O)ccc(-n2ccnn2)cc1 c1(NC(C2C(C)(C)C(NC(c3c[nH]c(C(N)=O)c3)=O)C2)=O)ccc(Cl)c(O)c1 c1(C(N(CC(C)NC(c2ccncc2C(F)F)=O)C)=O)cc2n(n1)CCOC2 Cc1nc2ncnn2cc1C(=O)NC1CCN(C(c2ccccc2O)=O)CC1O c1(SCC)cccnc1C(=O)NCC(C)(O)C(F)F C1(OCCNC(c2c(CC)ccs2)=O)CCN(C(=O)CCCOC)CC1 C1(NC(C2CCC(CC)O2)=O)CC2CCC1CN(C(=O)CSc1n[nH]c(C)n1)C2 Cc1ncsc1C(=O)NC1CCC1NC(c1cscc1Cl)=O.C1C(=O)N1 n1(CC(=O)NC(CC=C)CNC(=O)C(C(=O)OC)OC)nnc2ccccc2c1=O Cc1ccnc2sc(C(N3CCCN(C(=O)COC(C)(C)C)C(C)C3)=O)c(C)c12 c1(C(=O)OC)cc(C(=O)NC2CCCN(C(=O)C=Cc3cscn3)C2)cc(F)c1 c1(C(=O)NC2CN(C(CN(CC)CC)=O)CC(O)C2)cc(F)cc2nn(C)cc12 N1(C(c2c(C)cc(C)cc2O)=O)CC2CN(C(=O)CCn3cncn3)CC2(C)C1 c1(CC(=O)NC2CCCC(N(C(C(CC)OC)=O)C)C2)ccccc1C C1(C(=O)NCC(CNC(C(n2ccc(Br)n2)C)=O)(C)C)CCC2CC2CC1 CN1CC2CCN(C(c3ccn(CCNC(C4CS(=O)(=O)C4)=O)c3)=O)C2C1 C1(NC(=O)NC(CC=C)CC)CCC(C(C)C)CC1 CC1CN(C(c2csc(Cl)n2)=O)CC(C)CN1C(=O)CN1C(=O)CC(C)(C)C1=O c1(C(=O)NC(C)CCCNC(=O)C(c2ccccc2F)(C)F)ccc(Cl)nc1N c1(OC)ccc(Cl)c(C(=O)NC2CCCC2NC(c2coc(C(F)F)n2)=O)c1 C1(NC(c2c(CC)cc[nH]2)=O)CCCC(NC(=O)C(n2ccc(C)n2)C)C1 N1(CCC(N2CC(C(C)NC(C=CC(C)C)=O)C2)=O)CCCC1=O c1(C(C(=O)NCCOC)N(CC(C)OC)C(C)C)snc(OC)c1Cl C(C1=CCN(C)CC1)NC(CC1C(C)CN(C(=O)CC2CCCC(=O)N2)C1)=O CCC(C)CN=c1[nH]c(CC(=O)NOCCOC)cs1 C1(NC(C2=C(C)OCCS2)=O)CCCC2CN(C(c3ccc(=O)n(C)c3)=O)CC12 c1(C(=O)OC)cnc(CNC(=O)NCC(c2ccc(Br)s2)C)cn1 CCCC(C(O)C(=O)NC(C)CCN1CCCC1)NC(C1(C)CC(F)(F)C1)=O c1(C(=O)NC2CCCC(NC(c3c[nH]ccc3=O)=O)C2)cccc2nccn12 C1(C(=O)NCCOC(C)C)COCCN(C(c2cc(CO)ccn2)=O)C1 C(=O)(N(OC)C1CCC1)c1nc(CN(c2cc(C)nn2C)CC)oc1 C=CC1CCCN1C(CC1(C#N)CC1)C(=O)NCCOC.c12ccccc1N2 C12(NC(CC)=O)CCCC1CN(C(c1n[nH]cc1C1CCC1)=O)C2 CS(=O)c1ccc(CC(N2CCC3(C2)CN(C(=O)C2=CCCS2)C3)=O)cc1 C(=O)(N(CCC(=O)NCc1nccs1)OC)c1cccc(CC)c1 c1(C(=O)NCC2(C)CCN(C(c3cccs3)=O)C2)c(C2CC2)nc2sccn12 c1(C(N2CC(NC(c3cn(CC=C)nc3)=O)(CO)C2)=O)cccc(F)c1O N1(C(C2(C)ON=C(C)C2)=O)CCN2CCN(C(c3cn(C)[nH]c3=N)=O)CC2C1 C(CC(C)C)(C(=O)NC)NC(CC1N(C(c2nc(CC)oc2)=O)CC1)=O CCC(C)C(C)(O)CNC(C1CC(C)(NC(=O)C=CC2(C)COC2)C1)=O N1(c2cc(NCC3(C)COCCO3)nc(C)n2)CC2CC(C1)C2(C)C c1(C(N(C)SCC)=O)coc2c1CN(C(C1CC(C)C1)=O)C2 [N-]=[N+]=NC1CCC(C(=O)NC2CC3CCC2N(c2ncnc(=N)[nH]2)C3)CC1 c1(C(N2CCCC(NC(c3c[nH]cc(F)c3=O)=O)CC2)=O)cccc2cc[nH]c12 C1(NC(C(C2N(C(C(C)OC3CCCC3)=O)CCC2)(C)C)=O)CCOC(C)(C)C1 CC(C)(CCCNC(c1nn(-c2cccc(F)c2)c2c1CCC2)=O)C(=O)O N1(C(c2ccc(C)s2)=O)CC2CCN(C(=O)CC3CCC(C)(C)C3)C2C1 c1(CNC(C2N(C(C3C(C(=O)OC)C=C3)=O)CC2)=O)nc(NC(C)=O)cc(O)n1 C1(C(=O)NC2CCCC2)(CNC(CNC(=O)CC2COCCO2)=O)CC12CCC2 CC1CC(CNC(=O)CSc2nc[nH]n2)CN1C(=O)CC1CC2(CCC2)C1 N1(C(c2cc(CNC(=O)CC3CSC3)no2)=O)C2CCC1CC(CO)C2 CN1C(=O)CCCC1C(=O)NCC1CCCCCN1C(=O)C(c1ccccc1)=O Cc1c[nH]c2ncc(C(=O)NC(C(CO)C3CC3)C3CC3)cc12 CC1CCCCC1N(C(c1ccc(Cl)s1)=O)CC1(C)CN(C(=O)OC(C)(C)C)C1 c1(CNC(=O)NCCC2C=CCCC2)nc2ccccc2[nH]1 Cn1nc(C(=O)NCC2OCCC2C(=O)NC(C)(C)CF)cc1F Cc1cn(C)nc1C(=O)NC1CC(NC(c2n[nH]c(C(C)(C)C)n2)=O)CC1O CCCC(C(O)C(=O)NCCCc1cccnc1)NC(=O)CC(C)CCC N1(C(C(C)OC)=O)CC2C(CNC(=O)Cc3ccnn3C(C)C)C2C1 c1(NC(=O)NCCc2nn(C)nc2Br)ccc(F)c(Br)c1 CCC(O)C(C)(C)C(=O)NC1CC2CC1CN2C(=O)CCN1CCCC1 C(N=c1cc(C)nc(N2CC(=O)N3CCCC3C2)[nH]1)C1(Oc2cc(C)cc(C)c2)CC1 C(=O)(CC(C(C)(C)C)NC(=O)CCn1ccnn1)NC1(CSCC)CC1 C1(NC(CCCOCCC)=O)CC2CC(NC(=O)Cc3cnn(C(C)C)c3)CC12 C1(CC(=O)NCC(CCC)NC(c2ccc(C)c(CC)c2)=O)CCCC(F)(F)C1 c1(OC)ccc(C(N2CCC(F)(CNC(=O)Cc3ccccc3F)C2)=O)nc1 C1(CC#C)(NC(C2CC(=O)C2(C)C)=O)CCN(C(c2c[nH]nc2C2CC2)=O)C1 CC1=CCC(C(C)CC(=O)NCCSCc2cccnc2)CC1 c1(C(N2CCN(Cc3cc(O)c(O)c(O)c3)CC23CC3)=O)cc(Cl)cc(Br)c1Cl CCCCS(=O)(=O)CC(=O)NC1CN(C(=O)C(C)n2cnnn2)CC1C C1(NC(c2cn(CC)nc2C(C)C)=O)CCCN(C(=O)C=CC(=O)OCC)CC1F c1(CN(C)C(=O)NCc2cc(Br)no2)cc(-c2ccccc2)no1 Cc1cc(C(=O)NCC2CCN2C(=O)CSc2ccc(F)c(F)c2)c(C)c(C)c1 c1(OC)ccc(C(N2CCC(NC(c3csc(C)c3C)=O)C(F)C2)=O)c(OC)n1 CN=C(NC(c1ccc(C2CC2C)o1)C1CC1)NC1CC1C(F)F CCCCCC(O)CC(=O)NC(CNC(c1cnc(OC)cc1CC)=O)C1CC1 c12ccc(cc1)NC(=O)CNC2=O.n1(CCOC)cc(C2(N(C)C)CCC2)nn1 c1(C(c2n(CCC)nnn2)NCc2nc(C)co2)ccc(C#N)cc1OC N1(C(c2ccn(CCCC)n2)=O)CCC(F)(CNC(=O)C=NOC)C1 C1(C(N2CC(C(CC)C)C2)=O)CC12CCN(C(C1CC=CC(O)C1)=O)C2 C1(CC(=O)NC(C)CC(C)NC(C2CC(N(C)C)C2)=O)CC(O)C12CCC2 C1(CNC(c2ccc(OC)cn2)=O)CN(C(c2ccsc2OC)=O)CC(C)(C)C1 C1(C)(CCC(=O)NCC2(CNC(C(C)OCCC=C)=O)CCC2)CCC(=O)N1 CCCC(C(=O)N(C)C[Si](C)(C)C)NC(=O)CC(C)(C)OC N1(C(c2c(C)nn[nH]2)=O)C(CNC(=O)Cc2cn(C)nc2C)CC2CCCC12 c1(C(N2CC(C)(C)C(NC(C3CC(F)(F)CS3)=O)C2)=O)ccc2c[nH]nc2c1 N1(CC(COC)NC(=O)NCC2COC(=O)N2)CCOCC1 C1(C(=O)NC(C=C)C(F)(F)F)N(C(=O)C#CC(C)(C)O)CC12CCCC2 c1(C2(C(=O)NC(C(C)OCCOC)CO)CC2)ccc2c(c1)OCO2.C1C(=O)N1 N1(C(C(c2ccccc2F)C)=O)CC2(CC2)CC1CNC(C1CC2C=CC1O2)=O c1(C(=O)NCC2CN(C(C3CCCC3)=O)CCO2)cccc(O)c1Cl c1(C(CN(C(CC2CCN(CCCCC(=O)O)C2)=O)C)O)cccc(Cl)c1 Cn1nc(C2CC2)nc1C=O.N1CCCC(Cn2cc(C(O)C3CC3)nn2)C1 c1(C(=O)NC2(C(=O)NCC)CC2)cn(CCNC(C2(OC)CCC2)=O)nn1 c1(C(=O)NC(CC=C)CNC(c2c(C)[nH]c(C)c2C)=O)nccc2ccccc12 CCC(C(C)CN(C)C)NC(=O)C(C(C)C)NC(=O)CCc1nccn1C Cc1ccc2[nH]c(C(=O)NC(c3ncc(C)s3)C3CC3)cc2c1 c1(CNC(=O)OC)cn(C(C)CNC(=O)CNC(c2ccncc2)=O)nn1 CCS(=O)(=O)CC(=O)N(CCCNC(C1CC1c1ccc(Cl)cc1)=O)C1CC1 Cc1cc(-n2cccc2)ccc1C(N1CC(N(C(=O)C(C)O)C)C1)=O N(C1CCCc2ccoc21)C(c1cc(-c2ccc(C)cc2)[nH]n1)=O C1(NC(c2cc(C)ncn2)=O)CC2CC(NC(c3cn(C)cc3C)=O)C1C2 CC1CCC(C)(C(=O)NCCN(CCCN(C)C)C(=O)Cc2csc(S)n2)C1 C1(CNC(C(C=C)O)=O)(CO)CC12CCN(C(=O)C(F)(F)C=C)CC2 c1(C(N2CCC(NC(CCC(C)=O)=O)C(C)C2)=O)ccn2ncnc2c1 Cc1ccc(C(N2CCOC(CNC(C3CC3(C)C(C)C)=O)C2)=O)c(N)c1 c1(CN2CC3N(C(C4=C(C)OCC4)=O)C(C3)C2)c(C)cc(C)cc1C N1(C(CC2CCCC(=O)C2)=O)CCCC2C1CCCN2C(=O)Cc1cc[nH]n1 c1(CC(=O)NC2CN(C(CNC(CCOC)=O)=O)CC2C)n[nH]c2ccccc12 CC1(C)CC(=O)CCC1C(=O)NC1COCC1NC(c1cc(F)cc(Cl)c1)=O C1(CC(=O)Nc2n(C)ncc2-c2ccc(Br)cc2)CCCC2(CNC2)O1 Cc1c(C=CC(=O)Nc2nnc(-c3ccc(Cl)cc3Cl)s2)cnn1C c1(C(=O)NCC2(COC)CN(C(=O)CC3(N4CCCC4)CC3)C2)cc(C)ccc1C Cc1cc(N2CC3C(C)C3C2)nc(=NCCn2cc(C3CCOC3)cn2)[nH]1 N12Cc3ccccc3CC1C2.Cc1ccc(C(C)C)c(OCc2ccccc2)c1 C#CC1(NC(=O)C(CC2CCC2)NC(=O)OCC(C)(C)C)CCCOC1 C(=O)(C1CCCc2ncnn21)NCC(C(C)C)NC(c1c(C)c(F)ccc1N)=O C(=O)(C1CCc2cccnc21)NC(CNC(c1cccc(C)c1C(F)(F)F)=O)C N1(CCNC(=O)CN(C(=O)C(C2CCCCC2)F)CCO)CCC2CC12 Cc1ccc(C(N2CCC(C(C)NC(=O)CCN3CCNC(=O)C3)C2)=O)cc1C N1(C(C2(CC)CC(C)(C)C2)=O)CCCC(O)(CN(C)C(C2C=CCC2)=O)C1 Cc1ccc(F)c(CNc2cc(-c3cccc(C)n3)ccn2)c1 S(=O)(=O)(c1ccc(NCCS(C)(=O)=O)cc1Cl)N(C(c1cccc(Cl)c1)CO)C c1(C(=O)NCCC2CC(NC(C(C)OC(C)(C)C)=O)C2)ccc(OC(F)F)cn1 CCCCC(=O)N(CC(C)NC(=O)CN(C1CC1)CC)CC C1(CNC(C23CC(C(C)C)(C2)C3)=O)CCCN(C(c2ccc(N)cc2Cl)=O)CC1 C=CCC(C)(C)C(=O)NCC1CN(C(c2cc(C)n(C)n2)=O)C2CC12 C(=O)(CS(=O)(=O)C(C)C)NCC(CCCC)NC(=O)CCCOCCOC C(CCCCCNC(C1CCC(C)(C)C1)=O)NC(C(C)c1ccco1)=O Cc1ccc(C(N2CCN(C(C3CCC3(C)C)=O)C(CO)C2)=O)nc1O C1(CNC(=O)C=Cc2cncs2)CCCN(C(C2(CC3CCC3)CC2)=O)CC1 c1(C(N2CC(F)(CNC(C(C)(C3CC3)OC)=O)C2)=O)cccc(SC(F)(F)F)n1 Cc1ncnc(C(=O)NC(C)C(C)NC(=O)COc2ccccc2Br)c1C c1(C(=O)NC2CN(C(C=C(COC)C)=O)CC(O)C2)cc(OC)cc2c1CCC2 c1(C(C)C)ccccc1NC(c1cn(CCNC(C2CC23CCOC3)=O)cn1)=O N1(C(C(CO)NC(N)=O)=O)CC2CC2(CNC(=O)CCNC(=O)CO)C1 c1(C(=O)NCC2N(C(C(COC)(C)C)=O)CCCC2)cccc(OC)c1[N+](=O)[O-] c1(CC(=O)NC(CC)CN(C)C(C2CCNC2=O)=O)cc(C)ccc1F C(=O)(CC(C(F)F)NC(=O)C(C1CCCCC1)=O)NC(C(=O)OCC)C C1(NC(CC2ON=C(C)C2)=O)CCCC(NC(=O)C(C2CCCCC2)O)C1 N1(C(C(CCC)Cl)=O)CCOCC12CCN(C(C1CCCOC1)=O)C2 c1(C(=O)OC)c(OC)cncc1NC(C1CC(NC(c2cccnc2O)=O)C1)=O CCC(C)CCC(=O)N1CC(CNC(c2cccc(NC)n2)=O)(OC(C)C)C1 C(=O)(C(C)C(O)C(C)CC)NCC1CC(OC)CN1C(=O)C1=C(Cl)CCCC1 c1(CC)noc(C)c1C(=O)NC1CC(C)N(C(=O)C(F)(F)Oc2ccccc2)C1 c1(N(C)C)c(F)cc(CN2CC(F)CC2C(N2CCSCC2)=O)cc1F c1(OC)ccc(O)cc1NC(c1cc(CCNC(=O)CCC2CC(C)C2)on1)=O C1(CN(C(CCN(C(=O)C=C(C)C)CC=C)=O)CC)COCCO1 c1(NC(C(C)NC(C2CCN(CC)C2)=O)=O)ccc(Cl)cc1 C#Cc1cc(C(=O)NCCC2CCN(C(c3c[nH]c(=O)cn3)=O)C2)cc(Br)c1 C(=O)(C1=CCCCCC1)N1CCC(O)(C(C)NC(c2ccnn2CC2CC2)=O)C1 Cc1cc(OCC(=O)NCC(C)CN(C)C(c2ccsc2Cl)=O)no1 N1(C(C2(C(=O)OCC)CCCC2)=O)CCC(OCCOC2CC(C)N(C)C2)CC1 N1(C(C2N(C(COCCC)=O)CC2)=O)CC2CC1CS2 c1(NC(c2c(NC(c3c(OC)ccs3)=O)c[nH]n2)=O)cccnc1OC(F)F C(C1C(C(N2CC(NC(=O)C(F)C3CCOC3)CC2C)=O)C1(C)C)=C(C)C C=C(C)C1OCCCC1C(=O)NC1CCCC(NC(C2COCCN2C)=O)C1 CCC(C)(C(=O)N(CC(CO)(CO)NC(=O)C(C)C)C)OC c1(C2(C(N3CC(O)(CN(C(CC(C)SC)=O)C)C3)=O)CC2)c(C)cccc1C C1(C(C)C)CN(C(=O)Cc2ccsn2)CCN1C(=O)CN1CCCCS1(=O)=O c1(CNC(c2n(C(C(=O)OC)C)nnn2)c2sccc2Br)cnc(Br)c(F)c1 Cc1cc(C)c(S(=O)(=O)NC(=O)Cc2cc(C3CC3)on2)cc1[N+](=O)[O-] c1(CN2C(CNC(=O)OC(C)(C)C)CC2)ccc2cc(Br)ccc2n1 N1(C(=O)C2=CCC2)CCC2(CCCN(c3ncnc4cccc(F)c34)C2)C1 c1(C(N2CC(CC)(NC(c3cc(C(C)=O)oc3C)=O)C2)=O)c(C)ncn(C)c1=O C1(CNC(c2cc(CC)[nH]n2)=O)CN(C(=O)C(N2CCCC2)C2CC2)CC1(C)C C(=O)(C(CC(C)C)C(C)C)NC(CCC)CC(=O)NCC1NC(=O)NC1=O C(=O)(C(C)CS(C)(=O)=O)N1CC(CCC)N(C(=O)C=Cc2cnn(C)c2)CC1 c1(CCC(C)=O)cn(CC(C)NC(c2nc(C(C)(F)F)cs2)=O)nn1 C1(NC(C=CC(C)(C)NC(c2ccn(CCF)n2)=O)=O)CN(C)CCN(C)C1 C1(C)(CC=C)CN(C(=O)CNC(=O)CNC(=O)CC2CSCCO2)C1 Cc1nc(C(=O)NC2(CCO)CN(C(C3CCCC(N(C)C)C3)=O)C2)c(C)s1 c1(C(=O)NC2CCCC(CNC(c3c(OC)csc3)=O)C2)cc2n(c1)CCC2 c1(C(=O)Nc2onc(C(=O)OCC)c2C2CC2)ccc(S(C)(=O)=O)o1 C=C(C)CC(C)C(=O)N1CCN(C(c2cnn(C)c2)=O)C(CC)C1 CCS(=O)(=O)C1CN(C(=O)C(=O)NCCN2CCN(c3ccncc3F)CC2)C1 CC(F)(F)C(F)C(=O)NC1CCN(C(c2ccccn2)=O)CC1F N1(C(C2N(C(C)(C)C)CC2)=O)CCC2(CC1)CCN(C(C1CCCN1N=O)=O)C2 C1(C(=O)NCC2N(C(c3c(C)nc(C4CC4)o3)=O)CCCC2)CC2CC2CC1C C1(NC(C2CCC=CO2)=O)CCOC2(CCN(C(=O)C=CC=C(Cl)Cl)CC2)C1 N1(C2CCN(CCC=CCC)C2)CC(C)OC2(CCCOC2)C1 c1(NC=O)cnc(C2CC2)nc1.C12CC(C1)COCCC(=O)N2C.C1(N)CCC1 CCCC(C(=O)NCCN(C)C(c1ccsc1)=O)c1ccccc1 C1(CCOC)(NC(c2ccc(C(N)=O)o2)=O)CCN(C(C23C=CC(CC2)C3)=O)C1 c1(CS(N)(=O)=O)ccc(C(=O)NC2(CCNC(C3CCS(=O)(=O)N3)=O)CC2)cc1 CC1CCCC1(C)NC(c1ccn(CCNC(c2cncnc2)=O)c1)=O C1(OC)CCN(C(=O)CCCN(C)C(C2CCOC(=O)CC2)=O)C12CCC2 C(C)(C(C)C(=O)NCCOC1(C)CCC1)NC(c1nc(CC)oc1)=O CCCN=C(NCCc1cn2c(n1)SCC2)N1CC=C(F)C1 Cc1ccncc1C(c1nnnn1C1CC1)NC(C)CCN(C)C N1(C(C=CC(C)C)=O)CCCC1(C)C(N1CCCC(OC(C)C)C1)=O C1(C(=O)NCC(C(C)C)NC(=O)C(C)n2ccnc2)CN(CP(C)(C)=O)C1 C(=O)(C(C)CC(=O)OC)N1CC(C=C)(CC(N2CCN(CCOC)CC2)=O)C1 C1(C(N(CC(C)NC(C2(O)CCSCC2)=O)CC)=O)(OC)CCCCCC1 N1(C(CN(CC)CC)=O)CC(OC)CC1CNC(=O)C(C)n1cncn1 c1(C(=O)NCC2N(C(CCCC#C)=O)C3CCC2C3)ccc2c(c1)NC(=O)CS2 c1(C(=O)NC2CCC(N(C(CCNC(=O)OCC)=O)C)C2)c(F)cc(C)cc1F C1(C(N(C2CCCN(C(c3c[nH]nc3C(F)(F)F)=O)C2)CC)=O)CCCC(=O)N1 c1(C(=O)NC(C2CN(C(=O)CC3CC(C)(C)C3)CCO2)C)occ2c1CCCC2 c1(CNC(C2C3CN(Cc4cc(OC)ncc4Br)CC32)=O)cc(F)cc(C#N)c1 c1(NC(N2CCC(OCC(F)F)C2)=O)cc(N2CCOCC2)c(Cl)cc1Cl CC(C)(C)C#CC(=O)NCC1(C)CCN(C(C2COC(=O)O2)=O)C1 N1(C(Cc2c(C)nc[nH]2)=O)CCCC2C1CCCN2C(=O)CCCC(N)=O n1(CCNC(CCCNC(=O)OC)=O)cnc(C)c1C.C12(CC=CC1)C(=O)N2 C1(O)(CCC)CCN(C(C2CCC(CNC(c3cccn3CC)=O)CC2)=O)CC1 c1(N(CCOCCNC(C(C(C)C)NC(C)=O)=O)C)ncnc2c1CCO2 CC(CS(C)(=O)=O)C(=O)NCc1cn(CCNC(=O)C(C)(C)N(C)C)nn1 Oc1ccc(N2CCCCC2)cc1NC1COCC1CC1CCCCO1 C1(NC(C(CC)(C)O)=O)CC2(CCCN(C(=O)CN3CCC(C(N)=O)CC3)C2)C1 N1(C(=O)NC2(C(=O)O)C(C)CCC2)CCOC2(C1)CN(C(c1ccccc1)=O)C2 c1(C(=O)NC2(C(=O)NCc3cc(C)n(C)n3)CC2)ccc2cccnn12 c1(-n2c(-c3cc(C)sc3)nc(C3CC3)n2)cccc(S(C)(=O)=O)c1 C1(NC(C(C#C)(C)C)=O)CCN(C(=O)CCC(=O)c2cccnc2)CC1O CN1C(=O)CCc2cc(CNC(=O)CN3CCCC(OCC(F)F)C3)ccc21 CCC(CC)(C(=O)NC1CCCN(C(c2ccc(C)cc2OC)=O)C1)OC C1(CNC(C2(OCC)CCC2)=O)CN(C(c2ccnn2C)=O)CC12CC2 c1(NC(C2CC3CN(S(CC=C)(=O)=O)CC3C2)=O)cccc2c(O)nnc(O)c12 Cc1cc(F)cnc1C(=O)NC1(CCNC(=O)C(F)F)CCCC1 CC1C(NC(=O)Cc2ccccc2)CCCN1C(C1(C)OCCCO1)=O n1(CCNC(c2cc(CNC(C3CC=CC3)=O)[nH]n2)=O)ncccc1=O N1(C(CCc2c(C)noc2C)=O)CC(C(=O)Nc2cc(Br)ncc2F)C2(CC2)C1 C1(C(N2C(CC(=O)OC)CCC2)=O)COCCN(C(c2ncccn2)=O)C1 S(=O)(=O)(C1CCN(C(=O)NCc2nc(COC)cs2)C1)NC c1(N2CC(NC(=O)C(=O)NC3CCCCCCC3)(CO)C2)ncnc2cccnc12 C(C(=O)NCc1cccc(OC)c1)(C1=CCCSC1)N(CCC#C)C1CC1 c1(C(=O)NC2(CNC(C(CC)Cc3ccc(N)cc3)=O)CC2)cc(C)nc(C)n1 C1(C(=O)Nc2c(Cl)ncc(OC)c2)CCCC12CCN(Cc1cc(C)n(C)n1)C2 c1(C(=O)NC2C(CNC(C(CC=C)C)=O)CC2)cn(C)c2ncccc12 C1(C(=O)NCC2(C)CCCN(c3ncnc(C)c3Br)C2)CCC(C2CCCO2)O1 Cc1c(C(N2CCC3CCN(C(=O)C(C)(Cl)Cl)CC23)=O)ccc2n[nH]cc12 C1(C(=O)NC(C)CCN(C(=O)COCC(C)(C)C)C)CCCOC1 C1(CC=C)COCC1N=c1[nH]c(N2CCC(C)(N3CCC3)CC2)nc(=N)[nH]1 C1(n2cccn2)(CNC(=O)CC(F)F)CCN(C(=O)C(O)C2CCC2)CC1 C(N=c1nc(N(C)CCc2cn[nH]c2)c2cc(Cl)ccc2[nH]1)c1cn(C)[nH]c1=N Cc1cccc(OC(C)C(=O)NC2(CN)CC23CCC3)c1 N1(C(=O)NC(CC2CCC2)C(=O)NCCOc2ccncc2)CC2CCC1C2 N1(C(C(COC)NC(c2c(NC)cnnc2)=O)=O)CCCC(C)(C)C1C c1(C(C(=O)OCC)N(CC=C)CCN(C)C)ccc(C2CC2)c(F)c1 c1(CC)cccc(OCC(=O)NCCNC(=O)C(C)(C)C2CCCC2)c1 c1(OCC)ccc(C(N2CCC(NC(=O)C3=C(C)CCC3)C(O)C2)=O)cc1Cl C=C(F)C1(CC(=O)NCC(CNC(c2ccnc(C)c2)=O)CO)CCC1 N1(CC)CC(NC(C2CC=CCN2C(c2cncc(C)c2)=O)=O)C(C)(C)C1 C1(O)(C(=O)NC(C)C(c2ccccc2)NC(c2csc(Cl)n2)=O)CC(F)(F)C1 CN1C(=O)NCC1C(=O)NC1CCCC1(C)CNC(=O)CNC(N)=O Cc1ccc(N2CC(C(=O)N(CC(C)(F)C(C)(C)F)C(C)(C)C)CCC2=O)cc1C N1(C(CC2CC(NC(c3cnon3)=O)C2)=O)CCN2CCOCC2C1 C1(=CC(=O)N(C)CCNC(=O)CC(=O)Nc2ccc(O)cc2)CCCCC1(C)C C(C(=O)NCC1C=CCN1C(c1ccc(C#N)[nH]1)=O)(C(C)(C)C)N(C)C C(=O)(C(O)CC(F)(F)F)NCC(C1CCN(C(c2n[nH]c(C)c2Cl)=O)CC1)C N1(CCCCOC(C)C)CCC2(CC1)NC(=N)NC2=O N1(C(C(C)CN(C)C)=O)CC2(C(=O)NC3CN(C)C(=O)C34CC4)CCC1CC2 c1(C(=O)NC(CCCC)CNC(=O)CNS(=O)(=O)N(C)C)ccn2nncc2c1 N1(C(CCc2c(OC)cccc2)=O)CCCC2(C1)CC(OC)(OCC(F)(F)F)C2 C1(NC(C(C)Oc2ccc(Cl)cc2)=O)CC2CC1CN2C(=O)CC1(O)CCC1 C(=O)(C(C)(CNC(C1CCC(=O)CC1)=O)CC)NCC(CC)(C)C C1(N(C(=O)CC2CCCC(=O)N2)C)CCC2CN(C(C3CC=CC(O)C3)=O)CC12 CCC(C(=O)NCC(C)N(C(C1CC(F)CN1C)=O)CC)C(C)C c1(C(N2CCC(Br)CC2)=O)cc(-c2ccc(F)c(O)c2)cn2ccnc12 C1(C(=O)NCCCCCN(C(=O)CCn2ccnn2)C(C)C)CCCCC1F C(=O)(C1CCCc2ncnn21)NCC1(O)CN(C(C(C)(C)C2CCCCO2)=O)C1 C1(OCC)CN(C(C2(c3cc[nH]n3)CC2)=O)CC1CNC(c1cc(C)n(C)c1)=O S(=O)(=O)(c1cnc(C)c(C#N)c1)NCCCn1ncc(C)c1 Cc1cc(C(=O)NC(CC(F)F)C(=O)NCc2cc(C(C)C)no2)c(C)n1C CC1(C)CCC(CNC(=O)CC2(NC(=O)CC3CC=CCC3)CC2)O1 C1(NC(C(C)(C)OC)=O)CCCCC12CCN(C(=O)CSCCC(C)C)CC2 c1(C(=O)NC(CNC(c2c(C(=O)OC)c[nH]n2)=O)(C)C)ccc2c(c1)CCCS2 N1(C(C(C)OCCCC)=O)CCN(C(c2cnc(C(F)(F)F)s2)=O)CC1 C(=O)(CC(C)CC(=O)NC(C(=O)NCC1(C)CC2(CC2)C1)C1(C)CC1)OC C1(NC(Cc2ccc(C)o2)=O)CCN(C(=O)CCn2cc(Cl)cn2)CC1C c1(-c2cnc(C(C)C)[nH]2)nc(C2CCOC2)nn1C1CCCCCC1 CC1(C)OCCC1C(=O)NCc1ncc(C(N2CCCC2CCCO)=O)cn1 N1(CCC)CC2(CCC2)C1C1CCN(C(C2(COC(C)=O)CC2)=O)CC1 C1(C(N2CCC(N(C(c3cn(CCC)nn3)=O)CC)C2)=O)OCC2COCCC12 C1(NC(COC)=O)CCN(C(=O)CC2CCSCC2)CCC1(F)F Cc1cc(Br)cc(F)c1C(=O)NC1CCN(C(c2cnccc2C#N)=O)CC1O Cc1[nH][nH]c2ncnc(=NCC3CCCCC3Sc3ccccc3)c1-2 C1(NC(c2c(C)cc(OC)cc2F)=O)CN(C(=O)C=CSC)C2(CCOC2)C1 CC(C)CC(C(=O)NCCC1CCCN(C(c2cc(C#N)cs2)=O)CC1)C(C)C Cc1cc2ccccc2cc1C(N1CC(C)N(C(=O)C=CCO)CC1C)=O C12(C(N3CCC(CC=C)(NC(C4CCC(CC)CC4)=O)C3)=O)CCC(F)(CC1)CC2 c1(-n2c(C)ncc2)ccc(CNC(C2(C)CCCN2Cc2ccsc2)=O)cc1F C1(C(=O)NCC2(CN(C(c3c(CC)scn3)=O)C)CC2)CCCCCS1(=O)=O Cn1ccc(C(=O)NC2CCCC(NC(=O)CSc3n[nH]c(O)n3)C2)c(O)c1=O c1(C(N2C(CN(C(c3cc(CC)nn3C)=O)C)CCCC2)=O)cc(C)nc(C)c1 N1(CC(N2CCC(CC(=O)NC3(C4CCC4)CC3)C2)=O)CCOCC1=O CC1(CNC(c2nccnc2C(N)=O)=O)CCN(C(c2cc(O)nc(O)n2)=O)CC1 N1(C(C2(C(=O)OCC)CC2C)=O)CCC(CCNC(=O)CCCSC)C1 c1(C(=O)NC(CC)CNC(=O)C(F)(F)C2CCCC2)cc(S(N)(=O)=O)ccc1O c1(NC)ccc(C(=O)NC(C)(C)CNC(c2csnc2OC)=O)cc1 c1(C(N2CC=CC(NC(CC(CC)C(C)C)=O)C2)=O)cc(=O)c2ccccc2o1 C1(C)(C(=O)NC(CN(C(=O)CN2CSCC2=O)CC)C)COc2ccccc2O1 N1(C(CN(C(CN(C2CC2)CC)=O)CC2CC2)=O)CCCC(C(N)=O)C1 N1(C(C23CN(C(CCC(C)C)=O)C(C2)CO3)=O)CCC(C2(C)CC2)CC1 N1(C(C(CC)Cl)=O)CCC(O)C2(CCN(C(c3ccco3)=O)CC2)C1 c1(C(N2CCC(C)(CNC(C3CCCN3C=O)=O)C2)=O)noc2ccccc12 N1(C(c2c(C)ncs2)=O)CCCC(CN(C(=O)COc2ccc(F)nc2)C)C1 Cc1cc(C(N2CC3CC2C3NC(=O)C(O)C2CC2)=O)cc2nn[nH]c12 c1(OC)ccccc1C(C)CC(=O)NCCCCCN(C)C(c1sccc1F)=O N1(C(C(CC)=CCCC)=O)CCCC(NC(C2CC3CCC3C2)=O)C1 C1(C(=O)NCc2cc(C(N3CC(CC(=O)OC)C3)=O)n[nH]2)CCCCC1C C(=O)(C(F)(F)CO)NC(C1CCCCC1)C(=O)NC(c1nc(CC)on1)C N1(C(C2(C)CCN(C(C)=O)C2)=O)CCN(C(c2cccc(O)n2)=O)CC2(CC2)C1 CC(C)C(C)(CNC(=O)C(C1(C)CC1)NC(=O)C1=CCN(C)C1)C(C)C c1(C(=O)NCC(CNC(=O)C=Cc2ncco2)O)cc2c(o1)CCCNC2=O CC1(c2cn(C3(C(N)=O)CC3)nn2)CCN(C(=O)CC2CCCO2)C1 CCC(CC(=O)N(CCC(=O)NCCCN1CCOCC1)C(C)C)CC(C)C CCC(CC(F)(F)F)C(=O)NC1CN(C(C2(CN(C)C)CCCC2)=O)CC1OC c1(C(=O)NCC2N(C(C(C(C)C)C)=O)CC(O)C2)ccnc2ccsc12 Cn1cc(C(F)=CC(=O)NCC2CC2NC(C2CCC2)=O)cn1 S(=O)(=O)(c1cccnc1N1CCC2CCC(C1)N2C)N(C(C)CCO)C S(=O)(=O)(CCC(=O)N1CCC1NC(=O)C(=O)NCCOc1ccc(C)cc1)NC c1(C(=O)OCC)sc(-c2cccc(C(=O)N(C)Cc3cc(Br)co3)c2)nc1C c1(C(C(=O)NCc2cn(CC(C)NC(N)=O)nn2)O)cccc([N+](=O)[O-])c1 C1(NC(C23CC(CN(C(C=NOC)=O)C2)C3)=O)CC2CC1CC2(C)O c1(COC)cccc(NC(C23CC(C(N4CCC4(C)C(=O)OC)=O)(C2)C3)=O)c1 c1(C(=O)OC)c(NC(=O)N(C)Cc2cnc(C)s2)cnn1-c1ccc(F)cc1 n1(CC(=O)NCC2CC(NC(c3cnn(CCO)c3)=O)C2)cccnc1=O c1(CC(N2CCOCC2)C)cn(C2CCC(NCCO)C2)nn1 O=C(C1=NN(CCO)C(=O)CC1)NCC1CCCCN1C(C1(CO)COC1)=O c1(OC)ccc(C(=O)N(C(C)C(N2CCC(F)(CO)C2)=O)C2CC2)cn1 c1(C(N(C)CC2(NC(=O)CC3CCCC(C#N)C3)CC2)=O)c[nH]c2cccnc12 c1(OC)ccc(CC(=O)N(CC(C)NC(C2(CC(F)F)CCC2)=O)C)cc1F c1(CNC(c2ncc(C(C)(C)C)s2)c2nnnn2C2(C)CC2)ccc(Cl)cc1 c1(C(N2CCC(OC)C(F)C2)=O)ccc2c(c1)nnn2C C(=O)(CCCS(=O)(=O)N1CCOCC1)Nc1sc(C)c(C2CCCOC2)n1 Cc1nsc(C(=O)NC2CCCC2(C)NC(=O)C=CCCC(C)C)c1N c1(NC2CC(C)C(C)(C)CC2)cccc(S(=O)(=O)c2ccccc2)c1 NS(=O)(=O)CCC(N1C(CS(N2C(C(=O)OC(C)(C)C)CCC2)(=O)=O)CC1)=O n1(CC(=O)N(CC(C)NC(c2ccccc2CCN(C)C)=O)C)ncn(C)c1=O N1(C(C2N(C(CCn3ncc(C)c3)=O)C(C)CC2)=O)CC(=O)NCC1C(C)C c1(C(=O)NCC(CC)NC(=O)Cc2ccc(Cl)nc2)cc(C)nn1C c1(C(=O)NC2CC(OC)CN(C(C3CCO3)=O)C2)cc(F)cc2nn[nH]c12 C=CCC(C)(CO)CN=c1[nH]c(=N)[nH]c(=NCc2nnc(O)o2)[nH]1 c1(C(=O)NC2CC(CNC(c3c(CC)onc3C)=O)C2)ccc(Cl)c2occc12 c1(OC)ccc(Br)cc1C(c1nnnn1CCCF)NC1C=CCCC1 n1(CC(N2CCC(C3CCCCN3C(N3CCCC3)=O)C2)=O)ncc(O)nc1=O c1(N(C)CC2CCCN(C)C2)nc(=NCc2cn(C)nn2)[nH]c2ncn(C)c12 CCCC(N=c1[nH]c(=NC(C)c2cn[nH]c2)[nH]c2c1CSC2)C1CCC1 Cc1ccc(NC23CNCC2C3)cc1OCC(F)F Cc1cccc2c(C(=O)NCCCC(C)NC(=O)COc3ccsc3)n[nH]c12 C1(C(N(C)CC2CN(C(CCC(C)OC)=O)C2)=O)CC2(CC(C)=NO2)C1 c1(C(=O)NCCOCCCN(C(CCNC(C)=O)=O)C)cc2sc(C)cc2s1 c1(C(N2C(C(=O)Nc3nc(C)nc(O)c3)CC3CC32)=O)ccc(Cl)c(C)c1Cl C1(OC)CCC2CN(C(c3cc(Br)c(F)cn3)C(=O)NC3(C)CC3)CC12 c1(C(=O)NCC(C)N(C(=O)CCCN(C(C)C)C2CC2)CC)c(O)cccc1F c1(C(=O)NC2CCN(C(C(C)OCC#C)=O)C23CC3)ccc(Cl)c(Cl)c1C Cc1cn2c(n1)CC(C(=O)NCCC(C)(C)NC(=O)CC1OCCC1C)C2 C1(OC)CC(NC(=O)C=C2CCCC2)C12CCN(C(c1cc(Br)co1)=O)CC2 Cc1cc(C(=O)NCC2(NC(=O)C(CO)C(C)C)CCOCC2)c(N)c(Cl)c1 C1(CNC(C(CC)C#N)=O)CCCN(C(=O)COCCOCC)CC1 C1(NC(C2(CCC=C)CN(C(C3CCOC3(C)C)=O)C2)=O)CCCCCC1C c1(C(N2C(C(=O)NCC3(F)CCC3)CC3(CC3)C2)=O)cc(I)ccc1[N+](=O)[O-] N1(C2CCN(C(=O)NCc3sc(C)c(O)n3)C2)CC(C)OC(C)C1 c1(C(N2CCC(c3c(C)noc3C)C2)C(=O)NCC=C)cnc(OC)cn1 C1(C(N(C2C(C)CCN(C(C3(C(N)=O)CC3)=O)C2)C)=O)CCC12CCOCC2 c1(C(N(CCCNC(CCCN(CC)CC)=O)C)=O)ccc2nc(O)sc2c1 c1(C(=O)NCCOc2nncs2)cc2cc(F)c(F)cc2[nH]1 C1(CCNC(CC(C)(F)F)=O)CCCN(C(C2(CO)CCOC2)=O)CC1 c1(C(C(=O)NCC2CC2)N(CCOC(C)=O)C)ccc(-n2ccnc2)nc1 CC(C(=O)NCCC(Cc1ccccc1)NC(=O)CCn1ccnn1)S(N)(=O)=O N1(C(c2ccc(CNC(C(CC(=C)C)OC)=O)s2)=O)CC2(C)CC1CCO2 C(c1ccccc1Cl)=C(C(=O)NC(CCOC)CNC(C1CC=CCC1C)=O)C C1(CNC(CN(C)C2CC2)=O)CNCC1(F)CO.C1(C=O)CC1C(C)(F)F C1(C(=O)NCC2C3CN(C(Cc4nc(C(C)C)sc4)=O)CC32)CC(C)CC(=O)N1 C1(NC(c2nc(OCC)oc2)=O)CC2CN(C(=O)Cn3nnnc3C)CC12 N1(C(C2CC(C(=O)OC)C2)=O)CC(OC)C(NC(=O)C(C)C2CC2)C1 C1(CCOC)(NC(c2oc(C)cc2C)=O)CCN(c2nc(SC)ns2)CC1 C=Cn1nncc1C(N1CCC(CCN(C(=O)CC2CC3(CC3)CO2)C)CC1)=O CCCC(CC)C(=O)N1CCC(CCNC(=O)CCCC#N)C1 c1(C(=O)NC(CCN(C(Cc2cc(C)ns2)=O)C)C(C)C)cc(C)c(CO)cn1 C=CCC(F)(F)C(=O)NCCCN(C(=O)Cc1cccnc1Br)C(C)C C1(CNC(C2C(CCC)CCC2)=O)CC2CCC1N(C(C1(CC)CC1)=O)C2 Cc1ccncc1C=CC(=O)NCC(C)N(C)C(C1CC2(C1)CC2(F)F)=O C1(NC(c2ccnnc2)=O)CC(CO)N(C(C2CCCOC2)=O)C1 CCC(C)C(C)C(=O)NC(C1CCCN(Cc2cnc(C)o2)C1)C C1(CN(C(CSCCOC)=O)C)CCN(C(c2cc(-c3ccccc3)[nH]n2)=O)C1 C1(C(=O)NCC2CCSC2)C=CC(C(=O)NC2(C(O)CO)CC2)C1 C12(C(=O)NCC(CC(C)C)NC(CC(CC)C)=O)CCC(N(C)C)(CC1)CC2 c1(NC(C2(C)CN(C(=O)CCC3CC3)C2)=O)cn2ccnc2s1 Cc1ncn(C)c1C(=O)NC1CN(C(C2COCCN2C)=O)CC1C N1(C(C(C)(C2CC2)OC)=O)CC2CCC1CN2C(c1ncc(C)cc1O)=O C1(c2ccc(C)o2)COCCN1C(=O)NCc1cccc(Cl)n1 c1(NCC(CC)OC)nc2ccccc2nc1N(C)Cc1ncc(C)cn1 CCCC(C)(CC)C(=O)N1CCC(C2CCCN2C(=O)CC2CCC(C)CC2)C1 c1(C(N2CC(C)N(C(=O)CC(O)CC3CC3)CC2)=O)c(F)ccc(N)c1F CS(=O)(=NC(=O)C1NC2CC1CC2O)c1ccc(Cl)cc1 Cc1ncc(C(=O)NCCC(=O)NCc2ccc(Cl)o2)n1C N1(C(CCCn2cc(C(OC(=N)O)C3CC3)nn2)=O)CCCC(NC(N)=O)C1 c1(C(=O)NCCOC)cc(CN2CCC(C3OCCC(NC)C3)CC2)ccc1C N1(C(C2N(CC)CCC2)=O)C2CCC(C2)C1CC(=O)Nc1ccc(O)nc1 C(=O)(CC(C)C(=O)NC1CCCCC1CC(=O)NCCC1CCCCC1O)OC c1(CC(N2CC(CNC(C3CC(n4cccn4)C3)=O)C(O)C2)=O)ccc(Cl)c(Cl)c1 C#CC1(C(=O)NCCC2CC=CCC2)CN(C(=O)CCNC(=O)OCC)C1 c1(C(=O)NC(CNC(C2(SC)CCC2)=O)(C)C)ccc(Cl)cn1 C1(CCC=C)(C(=O)NCCOCCC=C)CN(C(C2CCC2(F)F)=O)C1 c1(C(=O)NC2C(C)CCN(C(C3(CO)CCC3)=O)C2)ccc2c(c1)C(=O)C(=O)N2 C1(C(=O)NCCCN(C(=O)Cc2ccsn2)CC)Cc2ccc(OC)nc2N1 C1(OC)CCN(C(=O)C(O)C2CN(C(=O)CN3CC4CCCC34)C2)C12CC2 C(=O)(CCCCC(N)=O)N1C(CNC(C2CC(C(=O)OC)C2)=O)C(C)(C)CC1 c1(C(N2CC(C)(C(F)(F)F)OCC2)=O)ccc2cc(Br)cnc2c1 Cc1nc(O)c(C(=O)N(CCC2CN(C(=O)C3CC3)C2)C2CC2)cc1C(F)(F)F N1(C(C(c2ccccc2)OC)=O)CCCCCC(NC(=O)C=CC=C(C)C)C1 c1(C(=O)NCCn2cc(CC(C)SCC)nn2)ccccc1S(=O)(=O)NC(C)C C1(CNC(C2N(C(C)=O)CC(O)C2)=O)CN(C(=O)C(O)C(C)C)CCN1C C(C(O)C(=O)N1CCC(C(C)(C)NC(c2cnc(CC3CC3)s2)=O)C1)=CC C1(CC)CN(C)CCN1C(C1CC(NC(c2cccc(CO)c2)=O)CCN1C)=O c1(N(C(C#C)=O)C(c2ccc(Cl)cn2)=O)ccc(SCC)cc1.C(CCCCC)N C12(NC(C(C=C)O)=O)CC1CN(C(=O)CCCNC(=O)OC(C)C)C2 N1(C(C2(C)CCCC2O)=O)CCC2(CC1)CNCc1ccccc1O2 S(=O)(=O)(c1ccc(Br)c(Cl)c1)CCN(C)CCN1CCOCC1(C)C CC1(C)CCC(C)(NC(C2CC3CCC(C2)N3C(=O)C=CC(F)(F)F)=O)CC1 C(=O)(CC(C)(C)c1ccccc1)NCC1N(C(C(CC)C2(C)CC2)=O)CC=C1 c1(CC(N2C(C(=O)NC3CCN(CCOC)C3)C=CC2)=O)cncc(C)c1 c1(CC(=O)NCC2N(C(C(=O)NC)=O)CC(C)(C)CC2)ccc(S(=O)C2CC2)cc1 Cc1cc2[nH]c(=O)c(C(N3CCC(N(C)C(c4cnc(S)n4C)=O)C3)=O)cn2n1 c1(C(N2CC3(C(NC(Cc4cc(C)nn4C)=O)CC3)C2)=O)cnc2c(c1)COC2 C1(C(N(CCC#C)CCO)=O)CN(C(c2sccc2C#N)=O)CC1(C)C C1(NC(c2c(COC)cc[nH]2)=O)CCN(C(=O)C(F)C2CCCC2)C1(C)C C(=O)(C(CC)C(C)(C)CC)NCCc1c(C(=O)NCCOCCCCC)c[nH]n1 C1(C(N(C)CC2OCCN(C(CCCOCCC)=O)C2)=O)CCc2c[nH]nc2C1 C(C(CC(F)(F)F)NC(=O)C(O)CN(C)C)NC(c1c(SC(C)C)cccc1)=O c1(C(=O)NCCC2N(C(C(C)O)=O)CCSC2)c(Cl)c2ccc(Cl)cc2n1C c1(C(N2CCC(C)(C(N(CCC(F)(F)F)CC)=O)C2)=O)ccc(C#N)c(C)c1 c1(C(=O)NCCCN(C(C2N(CCC)CCC2)=O)CC)cc(CO)ccc1Cl CCC(CC(=O)N1CCN(c2cccc(NC(=O)CCC3CC3)c2)CC1)C1CC1 Cc1ccc(C#N)cc1C(=O)NCC(CC(C)C)NC(c1ccnn1C(F)F)=O c1(CC(N2C(CN(C(C3CC(F)C3)=O)CC)CCC2)=O)cnccc1OC C1(N(C(c2nnn(C)n2)C(=O)NCC2CC2)C)C2CCOC2C1(C)C S(=O)(=O)(c1ccc2c(c1)CCO2)N1CCN(C(C(CC(C)C)O)=O)CC1CO N1(C(CC)C)CCN(c2nnc(CS(N)(=O)=O)n2CC2CC2)CC1 CN1CC=C(CCNC(=O)CC23CCC2CN(C(=O)C(O)C2CC2)C3)CC1 CC1CCC=C1C(=O)N1CCC1CC(=O)NCCCF C1(C(N2CC3(CCC(CNC(CN(C)C)=O)O3)C2)=O)COc2cc(O)ccc2C1 c1(C(N(CC(F)(F)F)C)=O)cc2n(n1)CCN(C(=O)CCc1ccccn1)C2 c1(C(N(CC(=O)O)Cc2cn(CCCCC=C)nn2)=O)cc2cccn2cn1 c1(C(N(C(C)C(N2CC(C)(C)CC2CO)=O)CC)=O)ccc([N+](=O)[O-])o1 CN(Cc1ccc(Cl)cc1)N1CCOC(CN(c2ccccc2)C)C1 N(C(=NCCF)N1CCC2=C(CCCC2)C1)Cc1c(C)ccc(C)n1 N1(C(CCOCCC)=O)CCCCC12CC(NC(C1CCc3n[nH]cc3C1)=O)C2 C1(CCNC(CCc2nc(C)sc2)=O)CN(C(c2ccc(F)o2)=O)CC1C N1(C(C(Cn2ccnn2)NC(C(CC=CC)C)=O)=O)CC(O)C(O)C1CO Cc1cccc(F)c1C(N1CCCC1C(N1CCC2(CC2)C1)=O)=O c1(C(=O)NCC(C)N(C)C(c2ccc(F)cc2N)=O)ccc(C#CC2CC2)cc1 C12CCC(C1)NC2=O.N1(C2CC(C(=O)NC3(c4nn[nH]n4)CC3)C2)CCOCC1 N1(C(CC(C)c2ccncc2)=O)CC2CC(C1)N2C(=O)CCC(C)(F)F Cc1ccc(C(=O)NC(C2CCN(C(c3cc(=O)cc[nH]3)=O)C2)C)c(F)c1Cl CC1(C(=O)NCC2CN(C(=O)CN3CCC(F)(F)C3)C2)CCCC1O c1(C(N2C(CNC(C=CC=CC)=O)CCC2)=O)ccc(OC)c(S(C)(=O)=O)c1 C(=O)(C(O)Cn1cncn1)N(CCN(C(=O)CCOC1CCOC1)C)C CC(C)CCC(F)C(=O)N1CCC(c2cn(-c3ccc(CCO)cc3)nn2)C1 N1(C(CC2(COC)CC2)=O)CCC2(CC(NC(c3cn(C)nc3C)=O)CO2)C1 N1(C(CCOCC#C)=O)CCN(C(=O)C(C)NC(N)=O)CC1CS(C)(=O)=O CC1(NC(c2ccnnc2)=O)CCN(C(C2(c3ccccc3)CCCC2)=O)C1 C1(NC(c2cccnc2SC(F)F)=O)CC2CN(C(C3CCCCC3)=O)CC12 C1(N(C(CCn2ccc(C)n2)=O)C)CCN(C(=O)Cc2ccncc2Cl)CC1C N1(C(CCN(C)CC)=O)CC2(C1)CN(C(C1(Cl)CCC1)=O)C2 C1(NC(c2cnnc(O)c2)=O)CC2CC(NC(C34CCCC3C4)=O)C1C2 C(C1=NOC(C)C1)NC(c1nc(C(C)NC(C2C(CC)C2)=O)oc1)=O Cc1cc(C(C(=O)NCCC2CC2)N(C2CC2C)C)c(F)c(Br)c1 c1(-n2cc(CCN3CCOCC3)nn2)nc(C2CC2)nn1CC1CCCOC1 C1(C(N(C(CCC(C)C)C)C)=O)CC12CCN(C(C1CC(N(C)C)C1)=O)CC2 CCCCCCC(=O)NC1CC1CNC(=O)COCC(=O)NCc1nc[nH]n1 Cc1cc2ccc(C(N3CC(NS(=O)(=O)C4CC4)CC(C)C3)=O)cc2[nH]1 C(CO)(CC(C)(C)C)NC(C1(NC(Cc2c(C)cccc2)=O)CC(F)(F)C1)=O c1(C(N2C(C(=O)NC(C=CC)C)CC2)=O)ccn(C2CC2)n1 N1(C(CC2CC(OCC)C2)=O)CCOC(CNC(c2cnccc2C)=O)C1 c1(N2CCCC(CC=C)(NC(C34CC(C)(C3)OC4C)=O)C2)cc(C)c(C#N)cn1 c1(CCC)nc(C)c(C(=O)NC2CCC(CN(C)C)C2)s1 N1(C(c2c(C)ccnc2C)C(=O)NCC)CCC2(COC(C)(C)OC2)C1 CC(C)CC(CNC(C1(C)CCOCC1)=O)C(=O)NC1(C2CCCC2)CC1 C1(C(=O)OC)(NC(=O)C2CCCC(=O)N2)CCCCC1.c1(N)ncn(C)n1.OC C(N=c1[nH]c2c(c(=NCc3cc(Cl)c(F)cc3F)[nH]1)COC2)C1(S(C)(=O)=O)CC1 c1(C(N(C2CCN(C(C3C(CC)C3)=O)C2)CC2CC2)=O)ccc(C)c(Br)c1N c1(C(N2CC(CNC(CC(COC)(C)C)=O)C(C)C2)=O)cc2c[nH]cnc-2n1 C1(O)(CCNC(C(C)c2ccon2)=O)CCCN(C(c2cc(Cl)c[nH]2)=O)C1 C(=O)(C1=C2CCCN=C2NN1)N(CCNC(C1CCC1(C)C)=O)CC c1(C(C(N2CC3C(n4cc(-c5cc(C)sc5)nn4)(C3)C2)=O)F)ccc(Cl)c(F)c1 C(=O)(C1Cc2ccccc21)NCC12CN(C(c3c(C)cccc3Cl)=O)C(C1)CO2 c1(C(=O)NCCN(C(CC2N(CC)CCC2)=O)C)ncccc1S(C)(=O)=O N1(C(C2(NC(CC3C(C)OCC3)=O)CCCC2)=O)CCN2CCC1C2 c1(CC)cc(N2CCC(NC(c3ccc(C(F)F)nc3)=O)C(O)C2)nc(C)n1 C1(NC(c2ccc(O)nc2)=O)CC(O)CN(C(C2CCCN2C2CC2)=O)C1 C12(NC(c3cncc(OC)n3)=O)CCC(C(=O)NC3CCCC(O)C3O)(CC1)C2 O=S1(=O)CCC2(CCN(S(=O)(=O)c3cc(F)c(F)c(F)c3)CCO2)C1 C1(C(=O)NCCOCC2CCOC2)CC2CCC1N2C(=O)C=Cc1cscn1 S(=O)(=O)(c1ccc(NC(C2(N(C3COC3)C)CCNCC2)=O)cc1Cl)N(C)C N1(C(CCS(C)=O)=O)CCC(C2(O)CCN(C(=O)CC3=CCCC3)C2)CC1 C1(NC(C(C(CC)C)C)=O)(CNC(=O)CNC(=O)NC2CC2)CC2CCC1CC2 C(C1=Cc2ccccc2OC1)=CC(=O)NC(C(C)C)(C)CNC(=O)C(O)CF N1(C(c2cc(C)[nH]n2)=O)CCN(C(=O)Nc2cccc(C3(C)CC3)c2)CC1 N1(C(c2c(C)nc(C)s2)=O)CC2CCC(C(N3CCCC3C3CCCC3)=O)(C2)C1 S(=O)(=O)(c1ccc(CC)c(Br)c1)N1CC(CC)CC1COCCCN(C1CC1)CC CCC(C)CC(=O)C(=O)N1CC2CC2(C(=O)NC2CC(O)CC2O)C1 C(=O)(C(C)(C)C(F)(F)F)NC(CNC(c1ccc(C)cc1N)=O)CC(C)C CCC(CC)(C(=O)NCC(c1ccccc1)NC(C1CCCNS1(=O)=O)=O)OC N1CCCCC1COCCN(C)Cc1noc(C2CC2)n1.C(C=O)OC c1(NC(CC(CC)NC(c2c(C)ccn2C)=O)=O)cc(O)ccc1C c1(C(=O)NC2CCN(C(=O)CC3CCC4CC4C3)C2)ccn(CCO)c(=O)c1 Cc1cc(C)c(C(=O)NC(C2CN(C(=O)CCCNC(N)=O)CCO2)C)c(C)c1 C1(C)(c2cc(OC)c(F)cc2)NC(=O)N(CC2=CCN(C(C)=O)CC2)C1=O O=C(CC1=NNC(=O)C1)NCCC1COCCN1C(c1ccc2cnsc2c1)=O N1(C(C(C(C)C)O)=O)CCN(C(C2(n3cnnn3)CC2)=O)C(C)C1 C(=O)(CC(C)C(=O)OC)NCC1(C)N(C(CCSCCCC)=O)CCC1 c1(C(=O)NCC2CC(O)(CNC(C3CCOC3)=O)C2)cc(F)cc2ccccc12 C1(NC(c2nc(CCC)oc2)=O)CCCN(C(c2c[nH]nc2CCC)=O)CCC1 CCCCCC(=O)N1CCC(=CCNC(c2cc(Br)n(C)n2)=O)CC1 c1(N2CCC(O)(C(C)NC(C3CCCC3C)=O)C2)ccnc(-c2nccs2)n1 c1(SCC(=O)N(CC(C)O)CCNC(CCSCC)=O)c(F)cccc1F C1(C(N2CC(c3cn(CC4CN(C(C(C)C)=O)C4)nn3)(O)C2)=O)CNC(=O)N1C c1(C(C)NC(=O)NC(c2nccs2)CC)ccc(OCC(F)F)cc1 c1(C(N2CC(NC(C3CCCC(C)(C)C3)=O)C2)=O)cc([N+](=O)[O-])c(F)cc1Cl N1(C(C(=Cc2ccco2)C)=O)CCC2CN(C(c3cc(C)c(C(N)=O)cn3)=O)CC12 c1(C(=O)NCC(CN(C(=O)C#CC2CCOC2)C)O)ccn2nccc2n1 N1(CCNC(=NCCC2(OC)CCC2)NCC2CCCS2)CCc2sccc2C1 c1(C(N(CCCNC(C(N2CC(C)C2)C)=O)CCO)=O)c[nH]cc1Br c1(CN2CCC(CC(=O)Nc3c[nH]ccc3=O)C2)cnc(Cl)c(F)c1 N1(C(C2N(C)CC2)=O)CCN2C(=O)C(NC(c3ccn4cccc4c3)=O)CC2C1 C(=O)(C1=C(Cl)CC1)N1C(CN(C(COC(CC)(C)C)=O)C)CCC1 C1(C(N2CCC(NC(c3c(C)nc(C)[nH]3)=O)C23CC3)=O)CC2C=CC1C21CC1 c1(OC)cncc(C=CC(N2CC3CCC3(NC(=O)Cc3nc(=N)[nH][nH]3)C2)=O)c1 C1(C)(CC)CN(C(=O)C(C2(C)CC2)N(C2CC2)CC)C1.c1(CCC=O)cnccn1 c1(OCC)cc(NC(C2CC3CC3N2c2ncnc3cc[nH]c23)=O)c(OC)cc1Br C(=O)(C1=CC(C)(C)C1)NCC(C)CN(C)C(C12CC(CO1)C2(C)C)=O N1(C(=O)NCc2cccc(C)c2)CCN(c2ccc(Cl)cc2C(N)=O)CC12CC2 c1(C(=O)NC(C(=O)N(C2CN(C(C=CCN(C)CC)=O)C2)C)C)ccccc1F Cn1cnc(C(=O)NCC2(CNC(=O)CCC3CCCOC3)CC2(F)F)c1 C1(C(N(C2CCCN(C(C=CC3N(C)CCC3)=O)C2)C)=O)CN2CCC1CC2 Cc1onc(Br)c1C(=O)NC1CCOCC1NC(c1ncc(F)cn1)=O c1(NC(C(CNC(=O)C(=O)NC2CC2)OC)=O)cc(CO)c(C)c(C)c1 C12(CC)CCCN(C1)C2=O.c1(NC(CCN(CCCCC)C)=O)cn(C)nc1C c1(C(C2CC2)NC(C(=O)N(CCC(F)(F)F)C)=O)ccnc(C(F)(F)F)c1 c1(C(=O)OCc2c(N=[N+]=[N-])cccc2)cnc2[nH]c(O)nc2c1 N1(C(C)C)C(=O)CCC1C(=O)NCC(=C1CN(C(=O)COCC2CCCC2)C1)F c1(C(=O)NCCOCCNC(CC(CC)(C)C)=O)c[nH]c2c(C)nccc2c1=O c1(C(C)OC)cn(CC2CCN2C(CC(C)C(F)F)=O)nn1 C1(C(=O)NCCCCNC(=O)C(C2CCCO2)C2CC2)CC2(CCCO2)C1 N1(C(c2ccnc(OC)c2Br)=O)CCC2(O)CCCCC2C1 C1(CCC)(NC(CC=CC)=O)CCN(C(c2cnn(CCO)c2CC)=O)C1 C(=O)(CC(C)(C)C#N)NCC(C(C)(C)C)NC(CC1CCCC(OC)C1)=O c1(C(=O)NC(CC)CNC(=O)C=Cc2ccc[nH]2)cc2c(Br)ccc(F)c2[nH]1 C=CC1(C(N2CCN(C)CC2)=O)CCN(C(c2cc(COC)on2)=O)C1 c1(COC)ccsc1C(N1CCCC1CNC(c1cc(-c2ccco2)cs1)=O)=O N1(C(c2c(CC)nccc2)C(=O)Nc2ccccc2)CC2(C(=O)O)CCC1CC2 CC1CN(c2ncc(F)cn2)CCC1CNC(=O)CCC1CCOCC1 C1(C(N2CCCC(CC(=O)OCC)C2)=O)Cc2ccc(Br)cc2C(=O)N1 C1(NC(CC)=O)COC2(CCN(C(c3csc(N4CCCCC4)n3)=O)C2)C1 C(=O)(C1CCCc2ccccc21)NC(C1(CNC(CSCC(C)C)=O)CC1)C c1(C(=O)NC2(C)CC(NC(C(C3CCC3)OC)=O)C2)cc(C(N)=O)cn1C c1(C(c2nnnn2CC)N)ccc(OC)c(F)c1.CCCCCC1CC1 N1(C(c2ccc(CNC(C)=O)s2)=O)CC2CCC1C(NC(c1oc(C)nc1C)=O)C2 c1(C(N2CC(N(C)C)CC(C(N)=O)C2)C(=O)NC)nn(C)c2c1CCC2 C(=O)(C1CCc2nccn21)NC(C1(C(=O)NC(C(C)C)c2ncc[nH]2)CC1)C C(=O)(C1CCc2ccccc21)NC1CCCC(NC(Cc2cn(C)nc2Cl)=O)C1 CC1CN(C(=O)C=CC(F)F)CC1CNC(C12CSCC1C2)=O C(CCC(C)(C)NC(c1ccc(C2CC2)cc1)=O)NC(CC1(C=C)CC1)=O C1(CN2CC(C#N)OCC2)CC2(CCOCC2)CO1 c1(NC(=O)C=CCSC)ccc(C)cc1.C(C(C)(C)CN1C(=O)C(=O)N1)OCC Cc1snnc1C(N1CCC(CCNC(c2ccsc2C(F)(F)F)=O)C1)=O C1(NC(C(c2cc(C)oc2C)C)=O)CN(C(=O)CS(C)(=O)=O)CCC1F Cc1cc(-c2ccnc(C(N3CCS(=O)CC3)=O)c2)c(F)cc1F C=CCC(CNC(=O)C(C)NC(=O)CCc1ccc(Cl)s1)NC(C1CCC1)=O C1(C(N(C2CCN(C(C3CCCC(=O)O3)=O)C2)CC)=O)CC(OC)C(OC)C1 Cc1sccc1C(=O)NC(C)(C)C(=O)NCC1(C#N)CC1 N1(C(CCCn2c(C)ncc2)=O)CC2CC1CN2C(=O)C=CC1CCCCCC1 C1(NC(C2ON=C(C)C2C)=O)CCCN(C(c2cccc(=O)o2)=O)C1C N1(C(c2c(C)c(F)ccc2)=O)CCOCC(F)(CNC(C2COCCO2)=O)C1 c1(CCC(=O)N(C(CCNC(CSCC)=O)C)C)ccc(F)c(OC)c1 C1(C(=O)NCC2CCC(F)C2)CCC(CO)CC1.C12(CC1)CCNC2=O N1(C(C=C(CCC)C)=O)CCC(C(C)(C)NC(=O)CCOCC2CC2)C1 N1(C(C2CCC(C)S2)=O)CCN(C(=O)Cc2c(F)cccc2C#N)CC(C)(C)C1 C(CS(=O)(=O)C(C)C)N(C(C(C)OCCC#C)=O)C(c1ccccc1F)=O c1(N2CCN(C(CCCC#C)=O)CC(O)C2)ncnc2c1nnn2C CC1(C)CCCN(C(c2cc(S(C)(=O)=O)co2)=O)C1CNC(C1CCSCC1)=O C1(C2CN(C(c3cnc(-c4ccsc4)s3)=O)C2)(NC(c2c(C)nc(C)[nH]2)=O)CC1 C1(C2CCCN(C(c3cnn(C)c(=O)c3)=O)C2)(NC(C2=CCC(C)CC2)=O)CC1 C(=O)(C(F)(F)C(O)C1CC1)NCC(C(C)C)NC(C1CC2(CSC2)C1)=O C(CC1=CCN(c2nccc(C#N)n2)CC1)NC(C=C(CC)CC)=O c1(CC(N2CC3CC(N4CC(F)C4)C2C3)=O)cc(C(F)(F)F)ccc1F N1(C(C(C)c2ccsn2)=O)CCC(O)(NC(=O)OC(C)(C)C)CC1 C1(CNC(CCc2c(C)ncs2)=O)CCCCN(C(c2ccc(O)nc2)=O)C1 C1(NC(CCOCCN(C(=O)C(F)(F)CO)C)=O)CCCCCC1CO N1(C(c2c(C)[nH]cc2)=O)CCC2(CCCN(C(=O)C(C)NC=O)C2)CC1 CC1(C)OCC2C(C(=O)NC3CN(C(C4CCS4(=O)=O)=O)C3)C2CO1 N1(C(c2c(CC)[nH]cc2)=O)CCC(C2CC(NC(=O)CCc3ccsc3)C2)C1 c1(C(=O)NCC2CC(C)N(C(c3cncs3)=O)C2)nc2ccccc2nc1O N1(C(C2(NC(c3c(C)non3)=O)CC(O)C2)=O)CC(=O)N2CCCC2C1 N1(C(CN(CCC)C)=O)CCOC2CN(C(=O)C3=CC(C)(CC)C3)CC12 N1(C(c2n(CC)ncc2C)C(=O)NC(C)C)CCOC(C(F)(F)F)(C2CC2)C1 N#Cc1cn(CCCNCc2c[nH]c3nccc(Br)c23)c(=O)nc1O C1(C)(NC(c2nc(C)sc2)=O)CCCN(C(c2c(C(C)C)cccc2C)=O)C1 NC1(C#CC(=O)N2CCC2C(F)(F)F)CCCC1 C(c1cc2ccccc2o1)=CC(N1CCN(C(C2CSC2)=O)CC1CO)=O c1(C2C(C(=O)NC3(CNC(CC(C)C)=O)CCCC3)C2)cccc(Br)c1 C1(C(N2CC(C(C(=O)NCc3cc(C4CC4)no3)OCC)C2)=O)CCCC(=O)CC1 c1(SC)ccc(C)c(C(=O)NCC2COC(CNC(=O)Cc3cncnc3)C2)c1 c1(C(C(=O)NCC(C)NC(=O)C(CC#N)C(C)(C)C)C)c(F)cccc1F c1(C(=O)NCC2N(C(c3cccc(CSC)c3)=O)CCC2)cnn2c1CCCN2 C1(NC(CC2(COC)CC2)=O)CC2CCC1CN2C(C1CCC(C)(O)CC1)=O c1(C(N2CC(C)(NC(C(CC)F)=O)C2)=O)ccc(C)cc1OC C1(O)(CC)CCC(NC(C2CCCCN2C(=O)CCC(C)(C)C)=O)CC1 CC1(C)COC(C(N2CCCCC(CNC(C3(CCF)CC3)=O)C2)=O)CO1 c1(C(=O)O)cc(Br)c(S(=O)(=O)NCC2CCC3(CCCCC3)O2)s1 c1(NCCCCS(C)=O)nc2ccccc2nc1NCc1ccc(Br)s1 CC1CCCCC1(CNC(c1cn(C)c(=O)n1C)=O)NC(=O)CC(C)(C)N(C)C C1(C(N2CCCC(CC)CC2)=O)C2CCN(C(C3(C)COCCO3)=O)CC12 N1(C(CC2(C)CCCCC2)=O)CC2CCC1C2NC(C1C(F)(F)C12CCC2)=O C=CCCCCCC(=O)NC1CCCN(C(c2cc(CC(C)C)c[nH]2)=O)C1CC C1(NC(C2C(C)CCOC2)=O)CN(C(=O)CSC2CCCCO2)C2CCCC12 C=C(C)C(C)(C)C(=O)NC1CCCC1NC(c1cnc(=N)[nH]c1)=O c1(OC)ccc(OC)c(-c2ccnc(O)c2CN2CCN(C)C(=O)C2)c1 c1(C(=O)NCC2C3CN(C(c4n(C)ncc4N)=O)CC32)cc2ccncc2s1 N1(C(c2ncc(C)c(Cl)c2)=O)CCCN(C(=O)CC#N)CC1c1ccccc1 C(CCC(=O)NCC(C)(C1CCC1)NC(=O)Cc1csc(NC=O)n1)C1C(C)C1 Cc1cc(Cl)ccc1OC(C)C(=O)NCC(F)CNC(c1cnc2n1CCC2)=O c1(CC)ccc(C(=O)NCC2CC3(CC(NC(=O)CC4CC(F)C4)C3)C2)c(C)c1 c1(C(Cn2cc(CNC(C=CCN(CC)CC)=O)nn2)C)cccc(F)c1 C(=O)(CC(CC)CC)N1C(C(=O)NC2C(CC)COC2)CCC1 N1(C(CC2(CSC)CC2)=O)CCC2(CCCC(CNC(=O)C(O)C(C)C)O2)CC1 C1(C(=O)NCCc2cccc(C)c2C)CC2C(=O)CCNC12 C1(=CC(=O)N2C3CCN(C3)C(=O)CC23CCC3)CCC(C)C1.CCO CCCC(CNC(C1(NC(C)=O)CCC1)=O)C(=O)N1CCC(C)(CO)CC1 N1(C(C2C(Cl)(C(=O)OC)C2)=O)CC(C2CN(C(c3nccc4n[nH]cc34)=O)C2)C1 c1(OC)cccc(OC)c1C(c1nnnn1CCCF)NCc1conc1C1CC1 C1(NC(c2c(C)cc(F)cn2)=O)CN(C(=O)C(C)N(C)C)C2(CCCCC2)C1 c1(C(=O)NC(CNC(C2(C=C)CCOCC2)=O)C)ccc2c(n1)NC(=O)CO2 N1(C(C(c2cccc(OC)c2)CC)=O)CCC(NC(=O)C=CCN(C)C)C(F)C1 C(=O)(C(O)CCCNC(C1(C(C)(C)O)CC1)=O)NC(C(C)O)C Cc1cc(C(N2CCCC2C(C)NC(c2ccsc2C)=O)=O)no1 O=C(CC1=CCOCC1)NC1CCCC1NC(c1ccc(C(F)(F)F)c(F)c1)=O C1(CNC(C2CCC(N(C)C)C2)=O)CC2(C1)CN(C(=O)Cc1nccn1C)C2 c1(CC)nn2c(c1C(=O)NC(C)CO)CCC2.c12cccc(c1)NCc1ccc-2s1 c1(C(CC(=O)NCC(C)NC(c2ncc(OC)cn2)=O)O)ccc(Cl)c(Cl)c1 CC1(C)CC(NC(c2ccn3nccc3n2)=O)CN(C(C2CCCC2)=O)C1 C(=O)(CCCCF)N1CC(=C(CNC(CC2(OC)CC2)=O)F)C1 N1(C(C2C(=C)C2)=O)CC=CC(C(N2CCC(COC)C2)=O)C1 C(=O)(CN=c1[nH]c(=NCCC(=O)N=c2cc[nH]cc2)[nH]c2c1CCC2)NCC c1(CC)nc(CC(=O)NC2CCCC2CNC(=O)C(CC)n2ccnc2)cs1 N1(C(CCCC(=O)OC)=O)CCC2CC2(C(N2CC(=O)N(C)C(=O)C2)=O)CC1 CCCCCCCC(=O)NC1CN(C(c2c(C)n[nH]c2C)=O)CC(F)(F)C1 N1(C(CCC(N)=O)=O)CC(NC(c2ncc[nH]c2=O)=O)CC(F)C1 C(=O)(CCC(CC)CCC)NC12CCCC(NC(C(CCC)C)=O)(C1)C2 c1(C(=O)NC(C(C)NC(=O)Cc2ccsc2)CO)cc(Cl)cc2c1NCCC2 C1(C(N(C2CCN(C(=O)CN(C)CCOC)C2)CCC)=O)CN2CCCC1C2 c1(C(=O)NC(C2CCN(C(=O)CCc3ccoc3)C2)C)cc(C2(C)CC2)on1 C(C)(C)(C(=O)N(CCCCCNC(=O)CCc1ccncn1)C)OCC C1(NC(c2cccc(NC)n2)=O)CCCN(C(=O)Cn2cnc([N+](=O)[O-])n2)CC1 C1(NC(C2CC(C)SCC2)=O)CN(C(C2(C#N)CC3(CC3)C2)=O)CC1(C)C N1(C(c2c(CC)ocn2)=O)CCN(C(C2(C(F)F)CC2(F)F)=O)CC1COC CCC(C#N)(CC)C(=O)N1CC(CNC(C2CC(C3CC3)C2)=O)C(F)(CO)C1 Cc1ccc(C(N2CCSCC2C(N2CC(O)(C(F)F)C2)=O)=O)c(F)c1 c1(NCC(=O)NCCCCC2CN(C(=O)C(O)CN3CCC3)C2)ccc(F)cc1 C1(C(=O)NCCNC(CC2ON=C(C)C2)=O)CC2(CCO2)C1 C1(C)(CNC(C2(CCCC)CC2)=O)CCN(C(C2(C)CC(C)C2)=O)C1 c1(C(=O)NC2C(CNC(c3cc(SC)oc3)=O)C2)cnccc1C(C)(C)C c1(CC)cc(C(N2CCOCC2CN(C(=O)CC=C(C)C)C)=O)oc1CC C12(C(N3CC(O)(CNC(C(C)SCCCC)=O)C3)=O)CCCC(=O)N1CCC2 CCC(C(F)(F)F)NC(=O)CC1(OC)CN(C(=O)CC2(COC)CCC2)C1 N1(C(C(CC)F)=O)Cc2cc(F)c(F)cc2C1 CC(C)C(O)C(C)C(=O)NC1CN(C(c2cnc(-c3ccccn3)s2)=O)CC1O C1(CNC(COC)=O)CC2(CCC2)CN1C(=O)C(C)(C)Oc1cc(F)cc(F)c1 N1(C(C2(CC#C)CC2)=O)CCC(CNC(=O)COC2CCCOC2)C(F)(F)CC1 CC(C)C(C)(CNC(=O)COc1cccc(F)c1)NC(=O)Cc1ccn(C)n1 N1(C(C(C2CC2)SC)=O)CCN(CCCNC(c2cc(C3CC3)on2)=O)CC1 C1(C(=O)NCC2(F)CN(C(CC3N(C(C)C)CCC3)=O)C2)CNC(=O)C(C)(C)C1 O=C(CC1C(=O)Nc2ccccc21)NCCOCCNC(C1CCCC1O)=O c1(C(N2CC(CNC(CN(C(C)C)C)=O)C(O)C2)=O)ncc(N)cc1Cl CC(=O)CCCC(=O)NCC1(F)CCCN(C(=O)C(F)=C2CCCC2)C1 N1(C(C2C3C=CSC23)=O)CCC2(CCCC2N2CC(F)(F)C2)CC1 c1(C(C)CC(=O)NC(C2(O)CN(C(C3CCN(C)C3)=O)C2)C)c(F)cccc1F CC(C)CC(C)(O)C(=O)NCCCC1CCCCN1C(=O)Cc1ccc(O)nc1 N1(C(CC2(CCC#C)OCCO2)=O)CCC(CNC(C2(C)CC3CC3C2)=O)CC1 c1(C(N2C(C)CCN(C(C3CCCC3O)=O)CC2)=O)ccc2c(c1)N(C)CCO2 CC1CCC(=CC(=O)NCC2(C)CCN(C(C3(CC(F)F)CCC3)=O)C2)CC1 c1(C(N(C(C(=O)NCC(=O)N(CC)CC)C)C)=O)ncc(C)cc1F C1(N(C(=O)C(Cc2ccc(O)cc2)OC(C)=O)CC)CCC(C(F)(F)F)N(C)C1 O=[N+]([O-])c1cnc2c(c1)CN(CC1CCC3(C1)CC3(F)F)CC2 C1(NC(CCCOCC=C)=O)CCN(C(c2nnn(C)c2C)=O)C1C(C)C N1(C(C2C(NC(C=CC=CC)=O)COC2)=O)CCC(C)CC1C c1(-c2cccc(OCCOC)c2)ccc2[nH]c(C(=O)NC3CNC(=O)C3)cc2n1 Cc1ccc(-c2ccc(C(=O)NCCCCNC(=O)CCCn3ccnn3)s2)o1 Cc1cnc2c(C(N3CCC4CN(C(C5CCCCN5C)=O)C4C3)=O)cccn12 CC(C)(C)C(CO)C(=O)NCCC1CCCN1C(=O)CCc1csc(=N)[nH]1 C(CS(=O)(=O)CC(=O)NC(C(=O)NCCC1CC1C(=O)OC)C1(C)CC1)OC c1(C(N2CC(C(N(C(=O)CCS(C)=O)C)=O)C2)=O)cc2ncc(Br)cn2n1 n1(CCNC(=O)OC(C)(C)C)cc(C(C(=O)NC2CC(C)C2)NC(C)=O)cn1 N1(C(c2cnc3n2CCC3)C(=O)NCCCSC)CCCOC(C(C)C)C1 C1(NC(c2c(C)coc2C2CC2)=O)CC2CCC(C1C)N2C(=O)CSCC(N)=O CCCCCCC(=O)NCC1(NC(=O)CSC2CC2)CC(F)(F)C1 O=C(CC(O)(C(F)(F)F)c1c[nH]c2ccccc12)N(CCCO)CCO C=CCN=C(NCCN1CCSCC1)N1CCC=C(c2ccccc2)C1 CCC(CCC(=O)NCCN(C(C)(C)C)CC)NC(c1ccncc1)=O N1(C(=O)OC(C)(C)C)CC(C2CCN(c3ccc(OC(F)F)cc3)C2)C1 Cc1ccn(CC(=O)NC2CN(C(=O)C(F)(F)c3ccccc3)CC2O)c(=O)c1 C1(CNC(CCC2CCN(C(CC=C(C)C)=O)C2)=O)NC(=O)NC1=O c1(C(=O)NCC2(C)N(C(CC3(C=C)CC3)=O)CCC2)cc(OC)c(N)c(C)c1 N1(CCC#C)CCC(C(=O)N(C2C3CN(C(C4CCCNC4=O)=O)CC23)C)CC1 c1(N(C(C2C(NC(COCC)=O)COC2)=O)CC)cc(F)ccc1OC c1(CN(C(=O)CS(C)(=O)=O)C)cccc(CNC(=O)CC2SC(=N)NC2=O)c1 CCCCCCCCCNC(=O)N(C)Cc1cn(C)nn1 c1(N(C)C)ccc(C(=O)NC23CC(C(=O)NCc4cnc(Cl)s4)(C2)C3)cc1 C(c1ccc(C(F)F)o1)=CC(=O)NCC(CNC(c1cc(CCOC)on1)=O)C c1(Nc2ccc(NC(=O)NC3CCN(C)C3)c(C#N)c2)ccc2ncc(C)n2c1 CC1CCN(C(C2(CCNC(C3C4CCC(F)(F)C34)=O)CCCC2)=O)CCS1 S(=O)(=O)(c1ccc(C(N2CCCC2)=O)cc1)N1CCN(CCN)C2C1C2 C1(CC(=O)NCC2(COC)CN(C(C(CC=C)C)=O)C2)CC(=O)NC(=O)C1 N12CCOCC1CC(=O)N1CC(C1)C(F)C2=O.C1(C(C)=O)CC(CC=O)C1.OC O=C(C#CC1CCC1)NCC1CCCCC1NC(c1c[nH]c(Br)c1)=O N1(C(C2C(C#C)C2(C)C)=O)CCCC2CN(C(c3csc(=NC)[nH]3)=O)CC12 c1(NC(C(CNC(C(F)=C(C)C)=O)O)=O)ccc(Cl)c(O)c1 c1(C(N2CCC3C(NC(CN(C(C)C)C)=O)C32)=O)ccc2ncc(Br)cc2c1 N1(C(c2c(C)cc[nH]2)=O)CCC2(CC1)CC(C(=O)Nc1cc(O)cc(O)c1)CO2 c1(C(N2C(CNC(=O)C3=CCCC3)CCC(C)(C)C2)=O)cc2c(Cl)nccc2o1 Cc1cnc(NCc2nccs2)c(S(=O)(=O)N(C2CCC(F)(F)C2)C)c1 Cc1ccc(C=CC(=O)N(CCC(C)NC(C2(CO)CCCO2)=O)C)o1 c1(C(N2CCC(C(CNC(C(CC)OC)=O)C)CC2)=O)cc2c(cc1O)CCC2 Cc1nn(CCO)cc1C(N1CCC12CN(C(=O)CCC(C)C#N)C2)=O Cc1nc2ccc(C(=O)NCCCC(=O)Nc3ccccc3)cc2[nH]1 c1(-n2cc(C(C)NC(=O)CCC3CC3(Cl)Cl)nn2)cccc(C(=O)O)c1 N1(C(C2CC(C)(CC)C2)=O)CCN(C(c2cc(Cl)ccc2Cl)=O)C(CCO)C1 CCCCC(CNC(c1cc(C2CCC2)on1)=O)NC(=O)CN1CC(C)(C)C1 CC(Cc1ccccc1)C(=O)NC1CCC(NC(=O)CCCN2CCCCC2)C1 c1(C(N2CCC(NC(C3CCCS3)=O)C(F)C2)=O)ccc2c(c1)OC(F)(F)O2 CON=Cc1ccc(C(N2CCN(C(=O)C(C)(C)CO)CC2CC2CC2)=O)cc1 c1(C(=O)NCCC(C)NC(=O)C2=NNC(=O)C2)cccc2ccnn12 c1(C(=O)NC(c2ccccc2)CNC(C(C)OC)=O)cnc(C)c(C)c1 Cn1cc(Cl)cc1C(=O)NCCC1(NC(=O)CC2CCC(F)(F)C2)CC1 N1(C(CCCc2scc(C)n2)=O)CCCCC1c1nc(=O)o[nH]1 C(CC(C(=O)NC1CCOCC1F)NC(c1n[nH]cc1C)=O)OC N1(C(c2c(C)cno2)=O)CC(CNC(=O)CCN(C)CCO)CC1(C)C c1(C(=O)NC2(CC=C)CN(C(=O)CCC3CC3)C2)cc(Cl)cn1C Cc1nc2c(C(=O)NC(C)CCNC(=O)Cc3cc(Cl)cc(Cl)c3)ccnc2[nH]1 CCC(CC(C)C)C(=O)NC1CN(C(c2cccc(OC(C)(C)C)n2)=O)C1 C=CC1CC(NC(c2coc(CNC(c3c[nH]nc3C)=O)c2)=O)C1 C1(O)(CNC(C(CCC)C)=O)CCN(C(C2(N(C)C)CCCSC2)=O)CC1 C=Cc1cc(C(N2CC(NC(=O)C=C(C)C(C)C)CC(F)C2)=O)cc(F)c1 C(CCCCC(=O)NCC1CC12CCCCC2)NC(COCC(=O)NC)=O N1(C(C2C(=C)C2)=O)CCC(COC)(NC(c2cccc(CN(C)C)c2)=O)CC1 C1(NC(C(CC)(CC)CO)=O)CCCN(C2CCc3c(F)cccc32)C1 CC1CCCN1CC(=O)N(C1CCCCC1)C(=O)CN(CCC(F)(F)F)C c1(C(N2CCCN(C(c3n[nH]c(C)c3Cl)=O)CC2C)=O)sc2nccnc2c1N c1(C(=O)NC(C(N2C(C)CC(C)(C)C2)=O)CC2CC2)cnn2cccc2c1 C1(N(C(CSC(C)C)=O)C)CN(C(c2ccc(C(F)(F)F)o2)=O)CCC1C CCC(C)(C)C(O)C(=O)N1CC2CC(NC(c3ccc(C)c(F)c3F)=O)C1C2 C1(C(=O)NC2CN(C(C3N(CC)CCC3)=O)CC2C(F)(F)F)CC(C)(C)CN1C CON(C(=O)CC1OCC(=O)N(C)C1c1ccccc1)C1CCCOc2ccc(C)cc21 C1(NC(CNC(=O)OC)=O)CC2CCC1(NC(=O)CC(C)O)C2 C1(NC(C2N(C(C34COCC3C4)=O)CCN(C)C2)=O)CCOC12CCCC2 N1(C(C2C(C(=O)OC)CC2)=O)CCN(C(=O)Cc2sccc2C)CC1C1CC1 c1(CCOC)nc(=NC(C(C)NC(c2cc(C(N)=O)ccn2)=O)C(C)C)s[nH]1 N1(C(C2(F)CCCN(C(CC3CCCC(C)O3)=O)C2)=O)CCC2(CCCC2)C1 c1(CCC(=O)NCCCCNC(C2(C(F)(F)F)CCC2)=O)c[nH]c2ccccc12 N1(C(C(C)OCC(C)C)=O)CC2(CNC(=O)CC3CC3)CCC1C2.c1ccccc1 c1(NC(C2CCN2Cc2ccncc2Cl)=O)c(Br)cc(F)c(F)c1F Cc1ccc(F)cc1CC(=O)NCC1CN(C(=O)C(O)C(F)(F)F)CCCO1 n1(CC(=O)NCC2N(C(COCCOC)=O)CCC2C)ncc2cccnc12 N1(C(c2c(C)cccc2)C(=O)NC2CCC2)CCc2c(F)cccc2C1 c1(C(=O)NCCCC2CCCN2C(C2CCC2)=O)cnc2c(c1)NC(=O)CO2 C1(C(=O)NCCSCc2n[nH]cc2F)CCCN(c2ccc(Cl)cc2Cl)C1=O C(=O)(C(O)CC(N)=O)N1CC(SC)C(N(C2CCC3(CC3)CO2)C)C1 C1(C(N(CCCNC(C2SCCCS2)=O)CCC)=O)CC2OC1C1CC21 c1(C(N2CC(OCC)C(CNC(=O)CC3CCCSC3)C2)=O)c(C)ccnc1O C1(O)(C(=O)NCCn2ncc(C(=O)NC(C#C)(C)C)c2)CCOC1(C)C C1(NC(CC(=C=C)C)=O)CCCN(C(c2ccc(NC)cc2Cl)=O)CC1 Cc1cncc(C(=O)NCC2COCCN2C(c2cccc(CN(C)C)c2)=O)c1 C1(CNC(CC2C(CC)C2(F)F)=O)CN(C(C2CC(O)CN2C)=O)CC1C c1(C(N(CCN(C(C2CC(CC)OCC2)=O)C)C)=O)cc(C)nc(Cl)c1N c1(CNC(=O)CC2(NC(c3ccc(F)c(I)c3)=O)CCC2)cc(Br)cc(Br)c1F c1(CCCC(=O)NCCn2cc(CCC3CCOC3)nn2)nc2ccccc2[nH]1 C1(C(=O)NC2C(NC(Cc3n(C(C)C)cnn3)=O)CCC2)CCC=CCC1 C12(CNC(c3ccc(F)c(Br)c3)=O)CCC1CN(C(=O)Cn1cnnn1)C2 N1(C(c2c(CC)n(C)cc2)=O)CC2ON=C(CNC(c3cnnn3C)=O)C2C1 CCCCC(C(=O)N1CCCC1C1(NC(c2cccc(C)c2Cl)=O)CC1)N(C)C N1(C(C)=O)CCCCC1C(=O)NCC1CCN(C(=O)CC2CCC(=O)N2C)C1 C1(NC(=O)CCc2cnco2)CCC2(CC1)CN(C(C1CC3CCC(C1)O3)=O)C2 Cc1ccc(C)c(Oc2ncc(O)cc2Cl)c1.c12cc(ccn1)NC(=O)NC2 c1(OC)ccc(CN(CCO)CC2(C(C)C)CCNCC2)cc1 C(=O)(CCCC(F)F)NC1C(CNC(C(C)SCC)=O)CCC1 N1(C(C2(CC)CC2(F)F)=O)CCN(C(c2cccc(C)c2)=O)C(C(F)F)C1 C#CC1(OCC(=O)NC2CCC2C(=O)NCC2(OC)CC2)COC1 C1(COC)CC(Cn2cc(CC(C)O)nn2)N(C(=O)Cc2ccoc2)C1 C1(NC(c2coc(Cl)n2)=O)C2CC3CN(C(=O)CNc4ccccn4)C1C3C2 c1(CN2CCCC(CN(CCCCCC=O)CCOC)C2)cc(C)c(Cl)c(C)c1 C1(COC)(CNC(C2CCSCC2)=O)CN(C(C2CC(n3cnnc3)C2)=O)C1 c1(C(=O)NC(CNC(c2onc(CC)c2C)=O)C2CCC2)c(C)cc(Cl)cc1N c1(C(=O)OC)ccc(C(=O)NCC(C2CC2)N(C(=O)C(C)(O)C2CCC2)C)nc1 C(C1CCN(C(=O)Cc2nc(=N)[nH][nH]2)CC1)=CC(=O)NCC(CC=C)(F)F c1(CC)ccc(C(=O)NCC2CC(C)(C)CN2C(C2CC(F)C2)=O)cc1[N+](=O)[O-] CCCC(C)(O)C(=O)NCC(C(C)(C)C)NC(c1cccc(F)c1NC(C)=O)=O C(=O)(CCCCC(F)(F)F)N1CCC(N(C(CC(C)(C)N(C)C)=O)C)CC1 C1(NC(=O)CCSc2ccccn2)CCN(C(c2cc3c(s2)CCC3)=O)CC1O C(CC(=O)NC1CCCCCCC1)(C(F)(F)F)NC(COCC(=C)C)=O C(CN=c1[nH]c2c(c(=NCc3cncc(F)c3)[nH]1)COC2)NS(=O)(=O)C1CC1 Cn1cc(CC(C(=O)O)NC(c2ccc3c(c2)CCCS3)=O)c2ccccc12 C1(c2n(CCCCCC)nnn2)(Nc2cnn(CCF)c2)CCSCC1 C1(NC(C(C)CC(N)=O)=O)CCCCCN(C(c2ccccc2N(C)C)=O)C1 c1(-c2cn(CS(C)(=O)=O)nc2)cnc2c(C(=O)NC3CCC(O)C3)c[nH]c2c1 c1(C(N(C2(C3CC3)CC2)C)=O)c(Cl)c(Cl)cc(Cl)c1Cl N1(CC2C(C)CCO2)CCCC1(C)COc1ccccc1 C(CCCCCC(=O)N1CCC(C)=C(F)C1)NC(C=C(C)C(F)F)=O N1(C(c2cc(C(=O)OC)no2)=O)CCC(C)(CNC(=O)COCCC(C)C)CC1 C12(NC(CCCOCC=C)=O)CCCC1CN(C(c1cnn3ccn(C)c13)=O)C2 N1(C(C2CC(=C)C2)=O)CC2CCC1C(NC(c1c(Cl)c(C)nn1C)=O)C2 CC1Cc2cc(C(N3CCC(NC(c4cnc(O)cc4O)=O)CC3)=O)ccc2O1 N1(C(c2cc[nH]c(=N)c2Cl)=O)C2CCC1C1CC1(NC(c1n[nH]cc1Cl)=O)C2 C1(C)(C(=O)NCC2N(C(CCCCCSC)=O)CC(O)C2)CCC(F)(F)CC1 c1(OC)cc(C(=O)NC(C)(CNC(=O)C(F)n2ccnc2)C(C)C)cc(Cl)n1 c1(NCC(C(=O)NC)C)cc(=NCC2CCC3(CCCC3)CC2)[nH]c(C)n1 N1(C(C(C)N2CCCC2)=O)CCN(C(=O)C(O)C2CC2)CC1c1ccccc1 c1(C(C(=O)OC)(C)NCC2CCCCC2N)ccc(F)cc1Cl c1(C(N2CC(O)(C(C)NC(c3c(C(C)C)nns3)=O)C2)=O)ccc(F)c(F)c1 C1(OC)(CNC(C23CC(CO2)C3)=O)CCN(C(c2ccsc2C#N)=O)CC1 N1(Cc2scc(C(C)NC(c3ncc(Cl)cc3Br)=O)n2)Cc2cccc(Br)c2C1 C(N=c1nc2ncn(C)c2c[nH]1)C1C(C)CN(C(c2cc3cscc3s2)=O)CC1 C1(C(=O)NCC(=C)Cl)CN(Cc2cc(CC)on2)CCO1 c1(NC(=O)NC2CCOCC2N2CCCC2)c(Cl)cccc1Cl C1(C(=O)NCC(C)=CC(=O)N(C)CC2COCCO2)CCC2(CCC2)O1 C(c1ccc(F)cc1F)=CC(N1C(C)CC(CNC(=O)CC2(C)OCCO2)C1)=O N1(C(C2CCC(=C)CC2)=O)CC2(CCCC2NC(c2ccc3cncn3c2)=O)C1 C1(NC(c2nc(C(N)=O)sc2)=O)CN(C(=O)COCC2CC2)C2(CCCC2)C1 N1(C(C2CN(C3CN(C)C3)C(=O)C2)=O)CCN(C(=O)CC2CCC2)CC(C)(F)C1 C1(NCCn2cccn2)C2CC3C(C2)C13C(N1CCCC1CCCO)=O.CC=O C(=O)(CCCCCn1cnnn1)N(C)CCn1cc(-c2ccc(Cl)nc2)nn1 c1(CC(N2CCN(C(CCOCC#C)=O)C(C)C2)=O)c(C)[nH]c2ccc(F)cc12 c1(N2CC3(C(NC(C(C=C)O)=O)CCS3)C2)nc(C(F)(F)F)c2ncnc-2[nH]1 c1(C(=O)NCCOC(C)C(N2CCNCC2)=O)cc(C(F)(F)F)ccc1CN c1(C(N2CC(N(C(c3nc(C(C)C)sc3)=O)C)C2)=O)csc(S(C)(=O)=O)c1 N1(C(c2c(C)non2)=O)CCC(F)CC1C(=O)NC1(n2cnnn2)CC1 N1(C(Cn2nnc(C)n2)=O)CCN(C(C2CCC2)=O)CC1c1ccc(F)cc1 CCCN=c1cc(C)[nH]c(=NCc2nc(C)cc(C)n2)[nH]1 c1(-c2nc(-c3ccc(C)o3)nn2CCOC(C)C)cnnc2ccccc12 CCC(CC(=O)N1CCC(NC(=O)COC(C)(C)CC)C(C)(C)C1)CC(F)(F)F C(C1NCCc2ccccc21)NC(c1ccccc1NC1CC1)=O C(CC(=O)NC1CCC12CN(C(c1ccnnc1)=O)C2)(C(F)(F)F)OC N1(C(Cc2c(C)ccnc2)=O)CC2(CNC(=O)C(O)C(C)C)CCC1CC2 C=CC(C)(CCOC)C(=O)NC1C2CC1N(C(c1coc(C(N)=O)c1)=O)C2 N(C(=NCC(=O)C1CC1)N1CCCC(OC2CCC2)C1)C(C)Cc1ccccc1 CC(O)CC(=O)NC(CNC(=O)C(C)NC=O)Cc1ccccc1 N1(C(CCCOCC=C)=O)CCN(C(=O)C(c2cccnc2)O)CC1C c1(C(=O)NC(COC)CNC(c2cscc2C2CC2)=O)ncc(Cl)cc1O C(=O)(CC(CC(C)C)NC(=O)CCS(C)(=O)=O)NC(CCC)(C)C N#CC1CCC(C(=O)NC2CC(c3cn(-c4c(F)cccc4F)nn3)C2)CC1 c1(C(CO)NC(C2CCOC(CN3CCCCC3)C2)=O)ccccc1I N1(C(C2CCN(C)C2)=O)CCN(C(c2csc(-c3ccsc3)n2)=O)CC1C(F)F c1(C(N2CC3C(NC(COCC(=O)OC)=O)(CC3)C2)=O)cccc2nccn12 CC(C)CN=C(NCC(O)Cn1cccn1)N1CCCC(C2(C)OCCO2)C1 c1(C(N2CCN(C(C3CCC(CO)CC3)=O)C(C3CCC3)C2)=O)n[nH]c2c1COC2 c1(C(N(C2CCN(C(=O)C(F)OC3CCOC3)CC2)C)=O)ccc(Cl)c(F)c1 c1(C(N2C3C(NC(CN(C4CCC4)C)=O)CC(C3)C2)=O)cc(N)c(Cl)c(O)c1 Cc1nc(C(N2CCCC2COC(C)(C)C)C(=O)NC2(C)CC2)c(Br)[nH]1 c12cccc(c1)C2.Cc1coc(-n2cc(-c3cnc(C4CC4)o3)nn2)n1 c1(N(C(C)C)C)ccc(C(=O)Nc2cccc(CC3CC(=O)NC3=O)c2)cn1 C=CCCCCCCCCC(=O)N1CC(O)(CNC(=O)C(C2CCCCC2)=O)C1 N1(C(CN(C(CCOCC#C)=O)CC)=O)CCC(CC)CC1 n1(CCC)cc(CC(C(=O)O)N(C(C)=O)CC)nn1 c1(OCC)ccc2c(c1)CC(C(=O)NCCN(C(=O)C=C(C)C(C)C)CC)CO2 N1(C(C=CSC)=O)CCCC(NC(=O)Cc2ccc(-n3cnnn3)cc2)C1C C1(NC(c2ccc(C(F)(F)F)s2)=O)CN(C(C2(O)CCOCC2)=O)CC1O C1(C(=O)OC)CCCCCN1Cc1nnc(N2CCCC2)o1 Cc1ccc(C(N2CCC(CNC(C3C(C#N)C3(C)C)=O)C2)=O)c(C(C)C)n1 C1(C(=O)NC2(CF)CCN(C(COC3(C)CCC3)=O)C2)CS(=O)(=O)CC12CC2 Cn1ccnc(CNC(CC(=O)OC(C)(C)C)c2ccccc2)c1=O c1(C(N2C(C(=O)NCc3ccc(SC)s3)CCC2)=O)nc2ccccc2[nH]1 C(=O)(C1CCCc2nccn21)NC1CC(CNC(=O)CN2CCCCCC2)C1 N1(C2(C(=O)NCCCN(C(=O)C=CCO)CCO)CCC2)CCOCC1 Cc1cc(C)c(C(=O)NCC2CC2NC(=O)Cn2cc(Br)ccc2=O)cn1 c1(C(=O)NC(C(C)C)C(C)NC(=O)Cc2cnccn2)cc(F)c(F)cc1N C1(C(N(C2CC(C(=O)NCC3(O)CCC(C)C3)C2)C)=O)CN(C)CCN1C C(=O)(CC(CC(C)C)NC(=O)C=C(C)c1ccco1)NC1CCCN(C(C)=O)C1 c1(NC(C(CO)NC(C(CC)CCOC)=O)=O)ccc2c(c1)CCC2 c1(C(=O)NCCOCCN(C(C(C)Cn2ccnc2)=O)C)cccc(CF)c1 C1(NC(Cc2ncc(CC)[nH]2)=O)CCN(C(=O)Cc2ccccc2F)CC1C c1(CNC2C(C(=O)NC(C(=O)OCC)C)C2)cc(Br)ccc1C Cc1ccc(C)c(C(=O)NC2CCN(C(c3cc(Cl)ncc3Cl)=O)C(C)C2)c1 CC1(F)CCN(C(c2sc(Br)cc2Cl)C(=O)NCc2ccccc2)C1 c1(C(N2C(CN(C(C(n3c(C)ccn3)C)=O)C)CCC2)=O)ccc(C(F)F)cc1 c1(C(=O)NC2CC(NC(c3ccnc(C)n3)=O)C(O)C2)c[nH]c2ccc(Cl)cc12 c1(CC(C(=O)N(CC(O)CC)CC#C)NC(=O)OC(C)(C)C)cccc(Br)c1 C1(C(=O)NC2CC(CNC(C3(C)CC=CCO3)=O)C2)CCS(=O)(=O)CC1 N1(C(C2(COC)CC=CC2)=O)CC(N(C(=O)C(=CC2CCCC2)C)C)C(C)(C)C1 C1(CC(=O)NC(C(=O)NCC)C)CCCC1NC(=O)C=CCOC C1(CNC(C(CC#C)(C)C)=O)(CO)CC12CCN(C(=O)C(C)NC(=O)NC)CC2 Cc1csc(Cl)c1C(=O)NCCOCCN(C)C(c1coc(C(C)(C)C)n1)=O N1(C(c2cc(=N)[nH]cc2)=O)CC(NC(=O)CCC2CC2(F)F)C2(CCCC2)C1 C(=O)(C1CCc2cccnc21)N1C(C#C)CN(C(c2ncn(C)n2)=O)CC1 C12(CNC(c3n(CC)ccn3)=O)CCCC1CN(C(=O)CCNC(C)=O)C2 C1(NC(c2csc(-c3ccc(Cl)s3)n2)=O)CCC(CNC(C2CC2CF)=O)C1 c1(C(=O)NCCNC(C2CC(CSC3CCCCO3)C2)=O)n[nH]c2c1COCC2 c1(CN(C(Cn2cc(C(C(C)C)N(C)C)nn2)=O)CCO)cncc(Cl)c1Cl C1(O)(CCNC(CC(CC)OC)=O)CCN(C(C2(CN(C)C)CC2)=O)CC1 N1(C(COCCCC#C)=O)CCCC2(CCN(C(C3CCCN3C(C)C)=O)C2)C1 C(c1ccc2c(c1)OCO2)=CC(=O)NC1CCN(C(c2scc(OC)c2)=O)C1 C1(SC)CN(C(=O)CCN(C)C(C)C)CC1NC(=O)C(C1CC1)C1CC1 CN1CCN(C(=O)CC2(C)CCOC2)CC1C(=O)NCc1ccnc(O)c1 CCC(CCc1ccccc1)C(=O)NC(C1(O)CN(C(=O)Cc2cnns2)C1)C CC(C)C(C)N=c1[nH]c(=NCc2ccc(N(C)C)nc2)[nH]c2ccccc12 c1(C(N2C3C(NC(CC=CCC)=O)CC(C3)C2)=O)cccc2c1NCCC2 C1(N(C(CSCC)=O)C)CCN(C(=O)C(C)OCc2ccncc2)CC1 c1(OC)nc(C(N2CCC(N(C)C(c3c(F)cccc3F)=O)CC2)=O)ncc1F C1(CNC(C2(CC#C)CC2)=O)CCC(C)N(C(C2CC2c2ccccc2)=O)C1 c1(OC)cc(C(=O)Nc2c(C(N)=O)ccnc2Cl)ncc1-c1cnn(CCF)c1 C1(F)(C(=O)OC)CCCN(C(=O)C(C)CN(C(=O)CCCOC(C)(C)C)C)C1 c1(CCC(=O)NCCNC(Cc2cc(C)nn2C)=O)cc(Br)ccc1Cl Cc1noc(C)c1C=CC(N1CCN(CCNC(=O)C(F)(F)CC2CC2)CC1)=O C1(CC)CC(O)CCN1C(=O)C(Cc1cnc[nH]1)NC(C1CCCC1O)=O c1(C(N2CCC(C)(CCNC(CCCCCC)=O)C2)=O)cc(O)ccc1[N+](=O)[O-] c1(SC)cscc1NC(=O)C(Cc1cnc[nH]1)NC(=O)OC(C)(C)C N1(C(C2C(C)C2(F)F)=O)CC2(CCCC2NC(c2cnc3cc[nH]c3c2)=O)C1 C1(C(=O)NC2(C)CCCN(C(c3n[nH]cc3F)=O)C2)Cc2cc(Br)ccc2O1 CC(CC(=O)N1CC2CC2(CNC(=O)CC2CSC2)C1)CC(C)(C)C Cc1nc(O)nc(C)c1CC(=O)NCC1COCC1NC(C1(C)CC=CCC1)=O c1(CCC(N2C(CNC(C3(C(C)C)CC3)=O)CCC2)=O)cccc(O)n1 CC(C)C1=NOC(C(=O)NCC2CCN(C(=O)COCc3nccs3)C2)C1 c1(C(N2CC3C(N(C(C(C)=CC4CC4)=O)C)C3C2)=O)c[nH]cc(Cl)c1=O C(=O)(CCCCCC(C)C)N1CC(O)(C(C(N2C(C(=O)NC)CC(C)C2)=O)F)C1 c1(SC)ccc(CCC(=O)N(CCCN(C(=O)C(=O)Nc2ncc[nH]2)C)C)cc1 CC1CN(C(C2CCNC(=O)C2)=O)CCN1C(=O)CN(C)CCO N1(C(c2cc(CCCCC)[nH]n2)=O)CCOCC1CNC(=O)CCc1cnoc1 C(C)(C(O)C(=O)NCCn1cncn1)OC.n12ccc(c1)C(=O)NCC2 C1(C(N2CC(C)(C)C2)=O)(OC)CCN(C(C2CCCN2C2CC2)=O)C1 Cc1nc(C(=O)NCC(Cc2ccoc2)CO)n2c1CCC2 N1(C(Cc2cc(OC)ncc2)=O)C2COCC1CC(NC(=O)C(C)(C)SC)C2 C1(NC(C(C#N)=CC(C)C)=O)C(C)CCN(C(c2ccc(F)c(Cl)c2)=O)C1C CC1CC2(CNC3CCN(C(c4ccco4)=O)C3)CC12 N1(C(C(=O)NCCON)c2csnn2)CCc2c(F)ccc(O)c2C1 C(=O)(C(O)CC[S+](C)C)N1CCC(CN(C(C(c2ccccc2)C)=O)C)CC1 C=CCCC(C)NC(=O)CNc1cn(-c2ccn(C)n2)nn1 c1(C(=O)NC2(C)CC(NC(c3cn(CCCC)nn3)=O)C2)ccc(C#N)s1 C(=O)(C(O)C(C)(C)C)N1CCC(C(C)NC(CCc2ccc(CC)cc2)=O)CC1 C1(CCC(=O)NC(C(C)(C)C)CO)CCCCN(C(=O)CC23CCCC2C3)C1 N1(C(CCCCNC(COC(C)C)=O)=O)CCCC12CCOC2=O C1(C(=O)Nc2cccc(-c3cnco3)c2)CC2(CC2)CN1C(c1nc(Br)cs1)=O CC(F)(F)CCCN=C(NCC1CCOC1)NC1CCCC1C(C)(C)C c1(C(c2ccccc2)CNC(N2CCC(OC)CC2)=O)nc2c([nH]1)CCCC2 c1(C(=O)NC2CC(C)CN(C(c3nc[nH]n3)=O)C2)c(F)ccc(Br)c1Cl c1(OC)ccc(C(c2nnc(N3CCC(OC)CC3)n2CCS(C)(=O)=O)=O)cc1 C(=O)(CCC(=O)c1cccs1)NCCC1CCN(C(c2ccn(C(C)C)n2)=O)C1 CC1CN(C(=O)CC(C)(C)n2cc(C(C)(C)F)nn2)CC1N(C1CC1)CC1CC1 C(C(=O)N1CC(CCO)(NC(=O)C(F)=C(C)C2CC2)C1)(C(C)C)SC c1(-c2ccc(C(N(C(C)CNC(=O)CCc3nncs3)C)=O)[nH]2)ccccc1F n1(CC)c(C(=O)N(CC(C)C(=O)N2CC(c3nncn3C)C2)C)cnc1O C1(CN(CC(C)O)C)CCN(C(C2CCCC2c2cnn(C)c2)=O)CC1 c1(N(CC(CN(C(C(COC)(C)C)=O)C)O)C)cc(C(F)(F)F)nc(Cl)n1 Cc1cc(C(=O)NCCN(C(c2occc2C2CC2)=O)C(C)C)c(O)c(C)c1 C1(CNC(C#CCNC(C(F)=C(C)C)=O)=O)NC(=O)CC1(C)C N1(C(C(CNC(C2C(C)SCCC2)=O)N(C)C)=O)CCCC(C)CC1 c1(OCC)cc(C(=O)N(CC(C)N(C(=O)CC(C)C(F)F)C)C)oc(=O)c1 CC(CCCC(=O)N1CCC(F)C1)NC(c1nc(=N)cc[nH]1)=O CC(C)CCC(C(=O)NCc1nn(C)cc1CC1CC1)NC(C1CC1(C)C(F)F)=O C1(CNC(C2C(C)(C(C)C)C2)=O)CCCCN(C(=O)CCc2ccco2)C1 C1(CC=C)(C(=O)NCC2=C(C)CCC2)CCN(C(=O)C(C)OCCN(C)C)C1 C#CC1(C(N2CCC(C(F)CNC(=O)C(CC=C)OC)CC2)=O)CCCC1 C(c1ccccc1)=CC(=O)N(CCNC(CC1C(CC)C1)=O)C C(=O)(CC1=CCCC1)N1CCC(CC(=O)N(C2CCSC2)C)C1 C(=O)(CC(C(F)F)NC(C1CCC1C)=O)NCc1c(CC)c[nH]n1 CCCCCCC(CC)C(=O)N(CCNC(c1n[nH]c(O)n1)=O)CCN(C)C c1(CC(=O)N(C2CCN(C(=O)CC(CC)C3CC3)C2)CCC)ccc(OC)cn1 C1(NC(C2(C)CCC(=O)N2)=O)CCCC(C(=O)NCC2CC(O)C(O)C2)CC1 N1(C(C=CC)=O)CCN(C(=O)CC2CCCN(C(C)C)C2)CC1c1cn[nH]c1 c1(OC)ncc(Cl)c(N(C(C)CCNC(c2cnc(O)nc2O)=O)C)n1 C1(C)(NC(CC(C)C2CC2)=O)CCC(NC(=O)CC2(N(C)C)CCCC2)CC1 N1(C(C)=O)CCC2CCN(C(=O)Cc3cc(Cl)ccc3OC)C2C1 C1(NC(CS(=O)(=O)NC)=O)CS(=O)(=O)C2CN(C(C3CCCN(CC)C3)=O)CC12 CCC(C)(C)C(=O)NC(CCc1ccccc1)C(C)NC(C1(C(C)C)CCC1)=O C(C)(CC(C)N=c1[nH]c2ccc(C(F)(F)F)cc2s1)NC(C(CC(CC)C)C)=O Cc1sc(S(N)(=O)=O)cc1C(=O)NCC(C)(C)CNC(C1CC(C)CC(C)C1)=O N1(C(c2cn(CCOCC)nc2)=O)CCN(C(=O)C2=C(C)CCC2)C(C)C1C C12(CC)CC(CN(CC(=O)NC(=O)CC)Cc3cccc(F)c3)(CO1)C2 N1(C(C(CC)C#N)=O)CC(CNC(=O)C(=Cc2ccccn2)C)CC(C)(C)C1 c1(C(N(C(C)CNC(=O)CCC2CCCC2)C)=O)c[nH]c2ccccc2c1=O N1(C(CCC(=C)Br)=O)CC2CCC1CN2C(=O)CCCc1nnc(C)n1C C1(C(N(CC#C)CCF)=O)CCN(C(C2CCC2(OC)OC)=O)C12CCC2 c1(C(N2C3C(CNC(C(CC)NC(C)=O)=O)C(C3)C2)=O)ccnc(Cl)c1F c1(-c2c(CN(C3CCCC3O)CCOC)csc2)ccc2c(c1)CCO2 C(C(C)C(F)C(=O)NC12CC(C1)C2)NC(C=Cc1ccc(C)o1)=O c1(CN(CCC(COC)OC)C=O)c(Cl)nc(Cl)n1C Cc1cc(C)c(C(=O)NCCCC(C)NC(c2ccnn2C(C)(C)C)=O)o1 C1(C)(NC(=O)NCc2cn(CC3OCCN(CC)C3)nn2)CCC(C)CC1 N(C(=NCCF)NCc1cccc(OC)c1OC)CCN(C)CC C(C1=NOC2CCCC12)Sc1ccc(-c2n(C(C)C)ncc2)nn1 C12(CNC(c3c(C)oc(Cl)n3)=O)CCCC1N(C(c1cncc(N)n1)=O)CCC2 c1(N)ccc(CO)cn1.Cc1cc(CN2CCC(C(C)C)C2)cs1.C12CC1CNC2=O Cc1cc(C(=O)NCC(C)(O)CNC(=O)CCn2c(C)ccc2C)sc1Cl c1(C(=O)NC2C(C(=O)NC(C(=O)NC)CC3CC3)CC=CC2)c(C)cccc1F c1(CC(=O)NC2CC(CNC(=O)CCC3CC3(F)F)C2)ccc2ccccc2c1 c1(C(C(N2CC(CNC(=O)CCOC3CC3)C2)=O)F)ccccc1 c1(C(C)(C)C)ccc(NC(c2nnnn2C2CCOCC2)c2ccoc2)cc1 Cc1nc(C(=O)NC(C2CCCN2C(=O)Cn2cnnn2)C)c2ccnc-2[nH]1 c1(CNC(=O)OC(C)C)cccc(C(=O)NCC2C3CCCOC23)c1 c1(C(=O)NC(CN(C(=O)Cc2cccc(Cl)c2)CC)C)c2c(nn1C)CCSC2 CCCCCCC(C)(CC)C(=O)N1CCC(C)(CNC(=O)CC2CC3CC3C2)C1 C#CCC(C)(C(=O)NC(C)CC(C)C(F)F)NC(c1ccnc(C)n1)=O N1(C(c2c(CC)onc2)=O)CCCC(N(C(=O)C(c2c(C)noc2C)C)C)CC1 CC1CCC(C(=O)NC2COCCC2NC(=O)COC2(C)CCCC2)CC1 C12(C(=O)N(CCn3cc(CN4CC5CC5C4)nn3)C3CC3)CC=CC(C1)OC2 N1(C(C(C)OCC(C)C)=O)CCC(NC(=O)CCc2ncccn2)C(CO)CC1 c1(C(=O)Nc2c(C#N)c(Br)cnc2)c(C(=O)NC2CC2)nn2ccccc12 C1(CC)(NC(c2ccccc2F)C)CCCOC1.C(=O)O C(=O)(C(C)CCO)N(CC(CN(C(C(C=C)O)=O)C)O)C c1(CNc2cc(N(C)C)ncn2)ccc(C(C)NC(C(C)C)=O)cc1 c1(C(CCCS(=O)(=O)N(C)C)c2n(CC)nnn2)ccc(F)c(OC)c1 N1(C(C2C3N(C(c4nc(C)c(F)cc4)=O)C(CC3)C2)=O)CC2CCN(C)CC2C1 CCCCS(=O)(=O)CC(=O)N1CC(NC(=O)C(c2cccc(F)c2)O)C1 c1(CC(=O)NC2C(CNC(C3(CC(C)C)CCC3)=O)C2)ccc(C(N)=O)nc1 c1(C(=O)NC(CC)CNC(=O)C(C)Cc2ccccc2)cc(N)nc(Br)c1 C=C(Cl)CCC(=O)N(C1CCC(NC(=O)CNC(c2cscn2)=O)CC1)C c1(N(C2CCC2)CC)ccc(C(=O)NOCC(C)O)cc1S(=O)(=O)N1CCNCC1 c1(C(=O)NCC2(CNC(C3C(C(=O)OC)CC3)=O)CCC2)sccc1C N1(C(c2c(C(C)C)occ2)=O)CC(NC(=O)CN2CCSCC2)CC2(CCC2)C1 CC1CC(CO)CN(C(C2(C3CC3)CN(C(=O)C(=O)C(C)(C)C)C2)=O)C1 c1(Cc2nc(-c3c(C)occ3)nn2CC(C)C2CC2)cc2cc(F)ccc2nn1 C(=O)(C(C)C(O)C(C)C)NC(C(N1CC(COC)CC(C)(C)C1)=O)C(C)C c1(C(C)(C)C)conc1C(=O)NOCC(=O)N(C1CC(CO)C1)C c1(CC(=O)NCC(C2CCC2)NC(C(C=C)(C)C)=O)csc2ccccc12 N1(C(c2cc(C)[nH]c2C)=O)CC(CNC(=O)C(c2ccc(F)cc2)C)CC1(C)C N1(C(CC(=C)C)=O)CCN(C(=O)CCNc2ccccn2)C(CC(F)F)C1 c1(C(=O)NC2CCCN(C(CC=C)=O)C2)cc[nH]c2nccc1-2 C(=O)(C1=CCCC1C)NCC(c1ccccc1OC)NC(CCOCC#C)=O N1(C(C23CC(OC)C2C3)=O)CCCC(NC(c2cn(C3CCCCC3)nn2)=O)C1 N(C1CCc2cccc(Br)c21)CC1CCC(C)(N2CCOCC2)CC1 Cc1cc(C(=O)NCC(C)N(C(=O)Cn2ccc(=N)[nH]2)C)nc(C)n1 Cc1nnc(CC(=O)NC2CC2CNC(=O)CNC(=O)CNC(C)=O)o1 C(CC(=O)Nc1cnc(OC)c(C)c1)(C(C)C)NC(c1nn(CC)c(O)c1)=O N1(C(C2C(=O)OCC2)=O)CC2CCC1CN2C(c1ccc2ccnn2c1)=O N1(C(C=CSC)=O)CC(NC(c2ccc(-c3nncn3C)cc2)=O)CC1C C1(NC(c2c(C)coc2)=O)CC(C)N(C(=O)CCC2CCC2)C1 C(=O)(C(C(C)(C)C)NC(=O)CC1OCCC1(C)C)NCC=CC(C)(C)C C(=O)(C(C(C)C)SC)NCC1(NC(C(CC)n2ccnc2)=O)CCCC1 c1(OCC(=O)N(C2CCN(C(=O)CCN3CCCC3)C2)C)cccnc1Cl c1(C(N(CC(C)NC(c2ccc(C#C)o2)=O)C)=O)ncc(OC)nc1OC c1(C(=O)NC2CC(C(=O)OCC)OCC2)c(C)sc(C)c1C#N C#CCCCC(=O)N(C1CC1)CC1CCCN1C(=O)C(O)Cc1cnc[nH]1 C1(CNC(C2(OC)CCC2)=O)CC2(CCN(C(c3cncc(C)c3)=O)C2)CO1 CCCC(O)CC(=O)N1CCOCC(CNC(=O)Cc2cncnc2)C1 C1(CNC(=O)Cc2ccn(C3CC3)n2)CCCCC12CCC2 C1(CNC(C(C)=C2CC2)=O)CC2(CCN(C(=O)C(C)(C)C(=O)N(C)C)CC2)CO1 c1(CC)ccc(C(N2CCC(CNC(C3CC3C3CC3)=O)CC2)=O)cc1Br C(CCC(C)(C)C(=O)N1CCCC(C)(O)C1)NC(C=C(C)C1CC1)=O N1(C(c2sccc2Cl)C(=O)NCC(=C)C)CCC(C2CCOCC2)(C(=O)OC)C1 C1(CC(=O)NCc2ccc(C(=O)NC3CC=CC3)s2)CCSCC1 c1(CNC(c2cnc(SC)o2)=O)cccc(CNC(c2n[nH]cc2C)=O)c1 N1(c2nc(C)cc(C(C)=O)n2)CCOC2(CCN(C(C34CC(C3)C4)=O)CC2)C1 Cc1ccc(C#N)c(N2CCC(NC(C3(C(C)C)COC3)=O)C(F)C2)n1 c1(CC)sc(C(=O)N(C2CCCN(C(=O)CNC(=O)CN(C)C)C2)CC)cc1C CC1(C)CC2(CO1)CN(C(C1CC(NC(C3CC4C=CC3O4)=O)CCO1)=O)C2 N1(C(C(C)OCCCC)=O)C(C(=O)NCc2ccnn2CC)CCC1C N1(C(C2(CCCC)CCCC2)=O)CCC(N(C(=O)CSS(C)(=O)=O)CCC)CC1 CC1CN(C(=O)OC(C)(C)C)CC1C(N1CC(NC(=O)C=C(Cl)Cl)C1)=O N(C(=NCCS(=O)c1ccccc1)NCCc1ccccc1)CC(C)C c1(CC)cccc(-c2nc(=S)n(COCc3ccc(Cl)cc3)[nH]2)c1 c1(CC)cc(CC(=O)NC2CCCC(NC(=O)Cc3cccnc3)C2)n(C)n1 c1(OC)c[nH]c(C(=O)NC2CCCC(NC(c3cn(C(F)F)cn3)=O)C2)cc1=O c1(OC)ccc(NC(C2C(O)CCN2C(c2cccc(O)n2)=O)=O)cc1I C(=O)(C(CC(N)=O)NC(=O)Cc1ncccc1C)OCc1nc(OCC)oc1 N1(C(C2(CC#C)CC=CCC2)=O)CCC(CNC(c2cscc2SC)=O)C(C)C1 N1(C(CSc2nc(C)[nH]n2)=O)CC(O)CC1CNC(=O)COC(C)(C)C C(=O)(CCS(N)(=O)=O)NC1CC(C)(NC(C2C(c3cn(C(C)C)nc3)C2)=O)C1 N1(c2cc(OC)ncn2)CC(C)(C)CCC1CNC(=O)CN(C)C(C)=O C1(CNC(C(F)=CCC)=O)CN(c2c(Cl)cccc2[N+](=O)[O-])CCC12CCOC2 CC1(C(=O)NCC(F)CNC(C2CN(C(N)=O)C2)=O)CCC(F)(F)CC1 N1(C(C2CC(n3ccnn3)C2)=O)CCCC(NC(C2(CO)CCC2)=O)C1 C1(C(=O)NCCCCCCNC(=O)C(F)C2CCOC2)CCC2(CC1)CC2(F)F C12(C(=O)NC(C)Cc3ccc(I)cc3)CCC(C1)C2(C)C c12ccnc(c1)NC2.c1(C(N)=O)csc(COC2CCCCC2)n1 c1(NC2(CNC(c3cn(C)nc3C(F)F)=O)COC2)nc2ccc(Cl)cc2s1 c1(C(N2CCN(C(C3CC(OC)C3)=O)C(C)C2C)=O)cc2ccncc2c(O)n1 C12(C(=O)NCCC(C(=O)NC(c3ncn(C)n3)C)OC)CCCC1OCC2 CC1CN(C(c2ccnc(C(F)(F)F)n2)=O)CC(C)N(C(=O)CC2(CO)CC2)C1 C1(C(=O)NC(C=CC(=O)NC(C#C)CC2CCCC2)C)CCCC(=O)N1C C1(C(C)(C)O)(CNC(c2ccnnc2)=O)CN(C(=O)CSC(F)(F)F)C1 CN1C(=O)CCC(C(=O)Nc2cc(F)cc(Br)c2F)C1c1cccnc1 C1(NC(=O)CSc2cccc[n+]2[O-])CN(C(c2cnc(C3CC3)o2)=O)C2CC12 c1(CNC(c2c(C(C)C)nco2)=O)cccc(CNC(C2CCC2C)=O)c1 C1(C(=O)NCCN(C(C)C)C(c2cc(Br)n(C)n2)=O)CC(=O)N(O)C1 c1(NC(C2C(C(=O)Nc3n(C)nc4c3CCC4)C2)=O)cc2ccc(Br)cc2s1 C(CC1c2ccccc2CCN1C(=O)CCSC(F)(F)F)NC(CCCCC)=O c1(C(N2CC(NC(C=C(CC)C)=O)C2)=O)nccc2cccnc12 CC(C)(CCCNC(=O)COCCCF)C(=O)NCc1cn(CCO)nn1 c1(C(=O)NCC(CN(C(CC(=O)NCC)=O)C)O)cccc2c1NCC2 C12(COC)CC(CNC(C3CC3C(N)=O)=O)(CN1C(C1CC13CC3)=O)C2 CC(CS(C)(=O)=O)C(=O)NCCC1(O)CN(C(c2ccc(F)c(C(F)F)c2)=O)C1 c1(C(=O)NCC(N2CCN(C(CS(CC)=O)=O)CC2)C(F)F)cccc(Cl)c1C CN1CCCCC1CC(=O)NCC1(F)CC(CNC(=O)CCn2cc(Cl)cn2)C1 c1(C(=O)NCC(COC)NC(c2c[nH]nc2C(C)C)=O)occc1C N12C(CCC1CC1CCN(C3CC3)CC1)C(=O)NCC2=O.C1(SC2CC2)CC1 C#CC1CCN(C(C2(O)CCN(C(c3cc(Cl)c[nH]3)=O)CC2)=O)CC1 c1(C(=O)NC(C(C)C)(C)CNC(=O)C(C)OCC(F)(F)F)cc([N+](=O)[O-])n[nH]1 c1(C(=O)OCC)c(N2CC3(CNC3)CCC2COC)nc2ccccc2c1C C1(NC(C(C)OC)=O)CN(C(c2cnn(CC)c2C2CC2)=O)CC12CCOCC2 c1(SCC(=O)N(CCCNC(=O)CN2CCCC2)C)ccc(F)c(F)c1 C(=O)(C(CCNC(C1(C)CCN(C)C1)=O)OC)NCCC(=O)NCC#C c1(C(=O)NCc2cn(C3CC(CSCC)C3)nn2)ccc(C)c(C(=O)OC)c1 c1(OCC(CN(S(=O)(=O)CCC(F)(F)F)CCCO)O)ccc2ccccc2c1 c1(C(=O)NCCCCNC(=O)C=CSc2nc[nH]n2)cc(Cl)c(O)c(Cl)c1 c1(CCC(=O)NCC2C3CN(C(c4c(=N)[nH]cnc4)=O)CC32)nnc(O)nc1O N1(C(C(C)C2CCCC2)=O)CC2(CC(NC(=O)C=CCN(C)C)CO2)C1 c1(NC(C(N2CCC(F)(CC)C2)=O)CCSC)ccc(S(N)(=O)=O)cc1NOC c1(C(N2CCCCC(C(=O)NCC3CC(C)(C)OC3)C2)=O)sccc1S(N)(=O)=O c1(C(=O)NC2(c3ccccc3)CN(C(C34CC(C3)C4)=O)C2)cc2n(n1)CCCO2 c1(C(=O)NC2CCN(C(c3cccc(Cl)n3)=O)CC2)cccc2cc(O)ccc12 c1(N2CC(C)S(=O)(=O)CC2)nc2c(c(=NC(C)c3nncn3C)[nH]1)COCC2 C1(NC(c2ccc(CO)cc2)=O)CCN(C(=O)C(F)(F)c2cn[nH]c2)CC1O C(c1nc(C)c(C)[nH]1)=CC(=O)Nc1cccc(NC(C(CC)OC)=O)c1 Cc1cc(C)n2nc(C(=O)NC(C3CCN(C(c4ccc(F)o4)=O)C3)C)nc2n1 C1(CNC(c2ccc(OC)s2)=O)CC(F)(F)CN1C(=O)CN1OC(C)(C)CC1=O c1(OC)ccc(C(=O)NC(CNC(=O)C(=O)CC(C)C)C2CC2)cc1Cl C(=O)(C1c2ccnn2CCN1C(=O)Nc1ccccc1OCCO)OC c1(C(C)(C)C)ccc(C(N2C3CN(C(=O)NC4CCC4)CC32)=O)cc1 C1(NC(CN(CCC)C(c2cscc2C#N)=O)=O)CC2OCCCC12 C(=O)(C1=C(F)CN(C(=O)CC2COCCO2)CC1)NC(CCCC=C)C CC1C(NC(=O)Cn2cc(Cl)cn2)CCCN1C(=O)C(F)C1CCC1 c1(COC)cccc(C(=O)NCCCCNC(C2(F)CCOCC2)=O)c1 N1(C(c2c(OC)n(C)nc2)=O)CCCC(C)C1CNC(c1oncc1C)=O C(=O)(C(F)C1=CCCCC1)N1CCCC(NC(c2cccn(O)c2=O)=O)CC1 N1(C(C(N2C(=O)CCC2=O)C)=O)CCC(C)N(C(=O)CC2C(C)(C)C2(C)C)CC1 CCC(C(=O)NC1CC(C(=O)NC(C)Cc2ccccn2)C1)NC(N)=O C(c1c(C)coc1C)=CC(=O)NC1CC(CCNC(C(CC)=CC)=O)C1 c1(C(=O)NCC2OCC(C)OC2)c(Cl)ccc(F)c1N CCCC(CC(=O)NC(C(F)F)C(C)(C)C)NC(=O)CN1CCC(C)C1 c1(C(=O)NCC(CC(F)(F)F)NC(CCCC=C)=O)cc(S(=O)(=O)NC)cs1 O=CN1CCOCC1C(=O)Nc1cccc(NC(c2ccc(Cl)o2)=O)c1 FCCCN=C(NC1CCN(CC(F)(F)F)C1)N1CCC(F)(c2cccc(Cl)c2)C1 N1(C(CN2C(C)CCC2)=O)CCC(C)(C)C1C(=O)NCC(F)CO C1(C(=O)NC2CCC(CNC(c3c(OC)cccc3)=O)C2)CC(=O)NC1(C)C N1(C(=O)COc2ccccc2)CC2(CCN2C(=O)CCc2ccccc2O)C1 C1(C(N2CCC(CNC(=O)CC3CCOC3)C(O)C2)=O)CCc2nc[nH]c2C1 N1(C(C(C)N2CCCC2)=O)CCN(C(c2cc(N)c(Cl)cn2)=O)C(C)C1 C1(NC(CNC(C(CC)C)=O)=O)C2CCCN(C(c3cc(C)no3)=O)C2C1(C)C c1(CN2CC(CNC(c3ccccc3)=O)C2)nnnn1CCc1ccccc1.CCN c1(SCC)cnccc1C(N1CCC(CF)(NC(=O)C(C)C2CCCC2)C1)=O N1(C(C2N(C(C3CC(N(C)C)C3)=O)CCC2)=O)CC2CCC1C(O)C2O c1(CNC(=O)CCC2CC2)c[nH]nc1C1CCN(C(=O)Cn2cccc2)C1 C1(NC(CCCOCC=C)=O)CCCC12CCCN(C(=O)COC(C)=O)C2 C1(C(N)=O)CCC(C(=O)NCCC2CCCN2c2nnnn2-c2ccccc2)O1 c1(C(=O)NC(CC)CNC(=O)Cn2nnc(-c3ccccc3)n2)cncc(C)n1 Cc1cc(C(N2CCC(NC(=O)C3=CCCC3)C(CO)CC2)=O)cn(C)c1=O Cc1oc(C2CC2)nc1C(=O)N(CCCn1cc(C(C)N(C)C)nn1)C c1(C(N2C(CNC(=O)COC3CCOCC3)CC2)=O)ccnc2ncnn12 c1(C(=O)NC(CC=C)CNC(c2ccnnc2)=O)cnn(CC)c1CC c1(Cc2n(CC)nc(-c3nccs3)n2)ccc2ncccc2c1 c1(C(=O)NCCCCCNC(CC2CC(CC)C2)=O)cnn2ccn(C)c12 C1(C(=O)NCCC(CNC(C2CC2C2CC2)=O)OC)CCC=CCCC1 Cc1cccc(C(=O)NCC2CC(NC(C3(C#N)CCC3)=O)C(O)C2)c1 CC1CCCN(C(=O)C=CCF)C1CCNC(=O)CCc1cccnc1Cl N1(C(C#CC)=O)C(CNC(=O)C(Cl)(Cl)Cl)CC2CC12 C1(CNC(C2C(C=C)C2)=O)(OC)CCN(C(c2csc(CC3CCC3)n2)=O)CC1 Cc1cccc(C(=O)NCCOc2cccnc2)c1C.c12ccnc(c1)C(=O)N2 C1(C(=O)OC)C=CCN1C(c1[nH]ccc1CNC(=O)COc1cccnc1)=O N1(C(CCSCCC)=O)CCC(C(F)CNC(c2ccc(COC)o2)=O)CC1 Cc1cc(C(=O)NC2CC(C(=O)NC3CCCC(O)C3)C2(C)C)c(C)s1 C1(C(=O)NC(C(C)NC(c2cn(CCC)nn2)=O)C)CC2(C1)CC1(CC1)C2 C1(C(=O)NC(C(=O)OC)C2CC2)(NC(COCC(=C)C)=O)CCSC1 CC(CCO)CCC(=O)N1CC(CNC(=O)C(O)C(F)(F)F)C2(CC2)C1 CCCC(CC(C)C)C(=O)NC1CC(C(=O)NCC(O)CN(C)C)=CC1O C1(C(N(CC(CNC(CSC)=O)O)C)=O)CC(c2cnn(C)c2)=NO1 c1(CNC(C(C)(N(C(=O)Cc2cc[nH]n2)C)C2CC2)=O)ccc(=O)n(C)c1 Cc1nc2ccc(C(=O)N(C3CN(C(=O)C(C(C)C)N(C)C)C3)C)cc2[nH]1 N1(C(C(C(C)C)O)=O)CCC2(CCN(Cc3ncccn3)C2)C1 C1(CCNC(C(C)OCCc2ccccc2)=O)CCN(c2ccccc2)C1=O O=C(C1=CCCCCC1)NC(C(=O)NC1(CC2CC2)CC1)C1CCC1 Cn1ccn2ncc(CNC(c3cn(CCN)cn3)=O)c12 C1(NC(C2CCCC(C)C2)=O)CCC2CN(C(=O)CC(C)(C)C)CC12 c1(C(N(CC(CNC(C(CC)OC)=O)(C)C)CC)=O)cnc(O)cc1OC C1(N(C)C)CCC(C(=O)NC2CCC(NC(=O)CN3CCCC3=O)C2)CC1 C1(C(N2C3C(C(=O)OC)C(C3)C2)=O)CC12CCN(C(=O)C=CC1CCCCC1)C2 c1(CNC(CC2OCCN(C(c3cc(OCC)ncc3)=O)C2)=O)ccc(Cl)cc1C CC1=C(C(=O)NC(CNC(=O)Cn2cnc(Br)c2)C(C)(C)C)CCS1(=O)=O C(=O)(C1=Cc2ccccc2C1)N1C(C)CC(CNC(c2ccccc2F)=O)CC1 CC(C)CCC(O)C(=O)N1CCC(CCC(=O)NC2CC(C)CC(C)C2)CC1 C1(C(N2CC3(CCN3C(C3CC4CCC3CC4)=O)C2)=O)(CC)CC2(CCC2)C1 CC(C)(C)C(C(=O)N1CC(O)CC1CNC(c1cccc(N)c1F)=O)C1CCC1 Cc1c(C(N2CCC(F)(CNC(=O)CC34COCC(C3)C4)C2)=O)cccc1F C1(CNC(=O)CCc2ccoc2)CN(C(=O)CCc2ncc[nH]2)CCC12CCC2 c1(C(=O)NC2CC3(C2)CC3Nc2ccc([N+](=O)[O-])cn2)cc2cc(F)ccc2[nH]1 C1(NC(C(CC)CC)=O)CC(C)CN(C(=O)CCCn2cncn2)C1 Cc1nc(=N)[nH]c(=NCC2CN(C(C3(C4CCC4)CCC3)=O)CCC2C)[nH]1 c1(CCNC(N(C2CC(F)(F)C2)CCCOC)=O)cn2cccnc2n1 N1(C(c2c(C)cc(CC)o2)=O)CCCC(NC(=O)CC2CCCOCC2)CC1 C1(c2n3cc(C)sc3nc2Cl)NC(=S)N(c2ccccc2)C2=C1C(=O)N(C)C2C c1(C(=O)NCC(CNC(C2(NC(=O)NC)CCCC2)=O)C)noc2c1CCCC2 C1(C(=O)NCC(CNC(=O)CCc2nc(CSC)no2)CO)(CC)CCOCC1 C1(CCCF)CCCC1(c1nnnn1CCCC1CC1)NCc1cccnc1Cl c1(C(N2CC3CCN(c4nccc(Br)n4)C3C2)=O)ccc2nc[nH]c2c1 N1(C(c2ccc(C(=O)OC)cn2)=O)CCCC(C2CC2NC(C2CC23CC3)=O)C1 N1(C(C(C)(C)CCCc2ccccc2)=O)CC(C2CCN(C(=O)CO)C2)C1 Cc1cc(C(N2CCC(O)C2C(=O)NCC2CCC(F)(F)C2)=O)cc(C#N)c1 C1(C(=O)NCc2coc(C)n2)(COC)CN(C(=O)CCc2cnco2)C1 c1(C(=O)NC2CC(NC(C3CCC(C#N)CC3)=O)C2)cc2c(Cl)cccc2s1 CC1=C(C(=O)NC2CCCCN(C(C3CN4CCC3CC4)=O)C2)CCCO1 C(=O)(C1=CCCC1(C)C)NC1(COC)CCN(C(c2cc(C)nn2C)=O)C1 c1(CC(N2CCC(COC)(NC(c3occc3F)=O)C2)=O)cccc(C)c1Cl C(=O)(C1CCCc2sccc21)NC1(C)CCCN(C(c2csc(C)c2N)=O)C1 c1(C(=O)NCC2CN(C(c3c(SCC)cncc3)=O)C2)cccc(C(N)=O)c1C N1(C(c2n(CC)cc(Cl)c2)=O)CCN(C(c2nnc(O)cc2O)=O)C(C)C1 CC1(C(=O)NCC=Cc2cccnc2)CCCN(c2nnc(C3CC3)n2CCO)C1 CC(C(=O)N1CCN(C(=O)COc2ccsc2Cl)C(c2ncc[nH]2)C1)C(C)(C)C c1(C2CCN(CC(=O)N(C(c3ccc(O)cc3)C(C)C)CCO)C2)ccc(Cl)cc1 N1(C(CCC)=O)CCN(C(C2CC(n3ccnn3)C2)=O)C(CO)C1 C1(C2CCN(C(=O)CC3CC4C=CC3C4)CC2)(NC(CC(CC)CC)=O)CC1 C1(N(C)C(C2CCCCC2)=O)CN(C(=O)CCc2ccc(O)cc2)CC12CC2 S(=O)(=O)(c1ccccc1NNC(=O)c1cc(=O)c2ccc(F)cc2o1)NC(C)C C1(C(=O)NC(c2cncs2)C)CSCN1C(=O)COC1CCCC1 C=CCC(CC=C)C(=O)N1CCC(NC(=O)CC2(O)CCCCCC2)C12CC2 C(=O)(CCN=c1[nH]ccs1)NC1CN(C(CCS(N)(=O)=O)=O)CC1C1CC1 CC1CCCCC1(C)C(N1CCC(F)(CNC(=O)CC2CCC2C)CC1)=O N1(C(C(C)(C)c2cnsc2)=O)CC2(CCC2NC(=O)CCCNC(=O)C2CC2)C1 N1(C(C(C)(F)F)=O)CCn2cc(C(=O)NCCOc3ccccn3)nc2C1 N1(C(c2c(CC)csc2)=O)CC2CCN(C(c3cccc(C)c3Cl)=O)C2C1 c1(-c2nc(CCC)nn2-c2cccc(F)c2)cc(C2CCCC2)nc(O)c1 N1(C(C2(C#C)CC2)=O)CCC2(CCC2CNC(c2cnn(CCO)c2C)=O)CC1 C(=O)(C(F)C(=O)N1CC(F)(C(=O)NC2CCN(C)C2=O)C1)OCC c1(C(N2CCC(C)C(NC(=O)COCC(F)F)C2)=O)ccc2c(c1)NC(=O)C2 CCCCCC(C)NC(C1(CNC(=O)CP(C)(C)=O)CC2(CC2)C1)=O N1(Cc2ccc(OCC)cc2O)CC2CN(C(=O)CCC3CC3)CC2C1 C(=O)(C1=CC2(CCOC2)C1)NC(C1(O)CN(C(C(CSC)O)=O)C1)C c1(CNC(NCCOC)=NCc2ccc(CO)cc2)ccc(F)c(S(N)(=O)=O)c1 c1(OC)ccccc1C(=O)NCc1cn(C2CCCC=C2Br)nn1 N1(C(C2(CC#C)CCOC2)=O)CC2CCC(C1)C2CNC(=O)C(C)(C)SC Cc1nc(=N)[nH]cc1C(N1CCCC1C(C)NC(=O)CCC1CCCCO1)=O CCC1=NOC(CC(=O)NC(C(=O)Nc2ccc(OCC)cc2)C2CCC2)C1 c1(C(N2C(C)(CNC(CCCC)=O)CCC2)=O)ccc(O)cc1O C(N=c1[nH]nc(C(N2CCC2C2CC2)=O)s1)c1c(C(=O)OC(C)(C)C)cccc1 C1(C(=O)NCCNC(=O)NCC)CC(C)(C)CN1C(C1C=C(C)CS1)=O c1(C(=O)NC(C(=O)NCC2CC2)C2CCCO2)cc[nH]c1 c1(N2CCCC(C=C)C2)nc(=NC)[nH]c(=NCc2cnc3c(Cl)cnn3c2)[nH]1 c1(C(=O)NCC(CCOC)NC(CCCCC=C)=O)cnc2sccn2c1=O c1(C(=O)NC2(CN(C)C(C3CCCC(=O)N3)=O)CC2)cc(Br)n(C)c1 N1(C(C#CC2(C)CC2)=O)CCN(C(C2(C(F)(F)F)CCCCO2)=O)CC12CCC2 CC1CN(C(c2cncc(CNC(=O)CCCC3CCCO3)c2)=O)CCC1O N1(C(C2(OC)CC(CF)C2)=O)CCC2C(C1)NC(=O)CN2C(=O)C=C(Cl)Cl C(CO)(CN=c1nc2scnc2c(NCC(c2ccccc2)N2CCCC2)[nH]1)OC N1(C(CCC(C)C)=O)CCCCC(CCC(N2CCOC(CN(C)C)C2)=O)C1 c1(C(N2CC(NC(c3c(SCC)nccn3)=O)C(O)C2)=O)cccc(Cl)c1F C1(NC(CCCN(C)C)=O)CC(C(=O)NC2CC3C=CC2C3)C1(C)C C1(NC(COc2c(C)cccc2)=O)CCCCN(C(=O)CSC(F)(F)F)C1 N1(C(C2CC(C)OCC2)=O)C2CCC1CN(C(=O)CNc1ncccn1)CC2 N1(C(c2c(OC)ccs2)=O)CCC(NC(=O)C(C)Cc2ccncc2)C1C1CC1 C(=O)(C(CCSC)NC(=O)OC(C)(C)C)NC1CC(NC(CC(=C)C)=O)C1 c1(C(=O)OC)cncc(C(=O)NC2CC(F)(CNC(=O)C(C)O)C2)c1C C(=O)(C(F)C(F)(F)C(F)(F)F)N1CC=CC(NC(=O)Cc2cocn2)C1 CCCCC(O)CC(=O)NC(C)(C)C(=O)NCC1(CO)CC=CC1 CCC(C)(F)C(=O)NC(C)CC1CCN(C(=O)CNC(N2CCCC2)=O)CC1 Cc1ccccc1C(C)(C)C(=O)N1CC(=C(F)CNC(C2(C)CS(=O)(=O)C2)=O)C1 N1(C(c2c(CC)nco2)=O)CCC(C)(CCn2cc(-c3ccc(C)nc3)nn2)C1 c1(CC(N2CC(O)(C(C)(C)NC(c3ccncc3)=O)C2)=O)cc(Cl)ccc1Br CC1(C)CN(C(=O)C(F)C(F)(F)F)CC1NC(c1csc(CO)n1)=O C#Cc1cnn(C)c1C(=O)NCC1CC1NC(=O)C(CC1CCCCC1)C(C)C Cc1nc(CCC(=O)NC2CN(C(C3CCC3)=O)CC2c2ccccc2)[nH]c1C N1(C(C2(C)CCCO2)=O)CC(O)(C2(CNC(c3cncc(F)c3)=O)CC2)C1 N1(C(CNC(CC)=O)=O)CCCC(C2(NC(c3ccc(=O)n(CC)c3)=O)CC2)C1 c1(OC)ccn2c(C(=O)N(CC(C)NC(=O)CCC3CC3C)C)cnc2c1 N1(C(CCCc2ncc(C)o2)=O)CCN(C(=O)Cn2cccn2)C(C)CC1C c1(CN2CCOCC(C(=O)NC(C(=O)OCC)C)C2)ccc2nc(O)[nH]c2c1 CCC(C)(C)C(O)C(=O)NCC1CC(C)N(C(=O)CC2(O)CCOCC2)C1 C1(O)(C(=O)NCC2C3CN(C(=O)Cn4cc(Cl)cn4)CC23)Cc2ccccc2C1 C1(CC(=O)N(CCC(=O)NCc2c(OC)scc2)CCO)CCCN(C)C1 C1(C(=O)NC2C(CC)CN(C(c3cccnc3F)=O)CC2)CCCCN(C)C1=O c1(OC)ccc2[nH]c(=NCCC3CCC(NC(c4cccnc4F)=O)C3)sc2c1 CC1(C)CC(NC(c2ccccc2Br)=O)CN1C(C1COCCO1)=O C1(NC(C=NOC)=O)CCC2(CC1)CCN(C(c1n[nH]c3ccc(Cl)cc13)=O)CC2 Cc1ccc(-n2nc(CCCN(C)C)nc2-c2cnc(C(F)F)s2)cc1F C1(C(N2CCC(CCNC(CC3C(CC)C3)=O)CC2)=O)CN2CCC1CC2.C1CC1 N1(C(CN(C(=O)CC(C)(C)C)CC(C)C)=O)CC(C)(C)C2COCC12 c1(C(N2C(C)CCC(NC(=O)CS(C)(=O)=O)C2)=O)ccc([N+](=O)[O-])cn1 C1(N(C(CCc2c(C)cccn2)=O)C)CCC2CN(C(c3oncc3C)=O)CC12 N1(C(C2C(OC)CCC2)=O)CCC(CF)(NC(C2CCOC2C(C)C)=O)C1 C1(NC(C2CC3(CCC3=O)C2)=O)CC2CC1CN(C(C1(CC3CCC3)CC1)=O)C2 Cc1noc(C)c1C(N1CC2C(CNC(c3cnc(C4CCC4)o3)=O)C2C1)=O c1(OC)cc(C(N2CCC(C(=O)NCc3cccn3C)C(O)C2)=O)ccc1I N1(C(c2c(SCC)cncc2)=O)CCCCC(N(C)C(c2ccnn2CC)=O)C1 c1(CC(=O)N(CCCCN(C(=O)CCc2cnoc2)C)C)cccc(F)c1O CC1COc2c(C(=O)NCC(O)CNC(=O)C(c3ccc(Cl)s3)C)cccc21 N1(C(C(C2CCOC2)OC)=O)CCN(C(C2CS(=O)(=O)C2)=O)CC(C)C1 C(=O)(C#CC1CCC1)NCC(CCNC(c1cncs1)=O)OC C(CCCCC(=O)NC1(C)CSC1)N(C)C(c1ncccc1O)=O c1(OC)ncnc(C(=O)N(C2CN(C(=O)CCCn3cccc3)CC2F)C)c1F CC1CCOCC1C(=O)NC1CC(CCNC(C23CC(F)(C2)C3)=O)C1 C1(NC(Cn2c(CCC)ncc2)=O)CCN(C(c2cnn(CCO)c2)=O)C1(C)C N1(C(CCCCC)=O)CCC(C)(CNC(=O)C2=NNC(=O)C2)CC1 N1(C(C2(OC)CCCC2)=O)CC2CC(CNC(C3C4CCCCC34)=O)C2C1 Cc1ncc(C(=O)NCC(CNC(C2CC23CCCCC3)=O)CO)c(C)n1 C12(C(=O)NCC(CNC(CCCC(=O)N(C)C)=O)(C)C)COCC1CS(=O)(=O)C2 CON1CCC(CC(=O)NCC2(C)CCCN2C(c2sccc2F)=O)CC1 CC(Cn1cccn1)C(=O)N(C(C)(C(=O)N(C)CC1(N(C)C)CCC1)C1CC1)C C1(O)(C(=O)NC(C)CNC(=O)C(O)C2CCC2)CCCC(C)(C)C1 C1(COC(C(=C)CCNC(=O)OC(C)(C)C)=O)CCC2CN(C)CC2C1 C(N=c1cc(Cl)nc[nH]1)C1CC(C)N(C(C2Cc3cscc3C2)=O)C1 N1(C(C(C)(CC2CCC2)OC)=O)CCC(C2CCN(C(=O)C(N)=O)C2)CC1 CCCCCCC(C)(CC)C(=O)N1CCN(C(=O)C(C)=C2CCC2)C(C(F)F)C1 Nc1nc(C(=O)NCC2(NC(=O)Cc3ccccc3Cl)CCC2)ccc1O Cc1cc(C(=O)NCC(C(C)(C)C)NC(C2(C)CC2C)=O)nn1C1CC1 CCCCC(C(=O)N1CC2(CCN2C(=O)CCC2C(=O)NN=C2C)C1)N(C)C C1(C(=O)NC(Cc2ccc(O)cc2)CO)CC(F)CN(C(=O)C=CCBr)C1 c1(C(=O)OC)cnc(NC2CC3CN(C(=O)C(C)SC(F)(F)F)CC23)c(Cl)c1 c1(-c2cn(CC3N(C(C(CCOC)(C)C)=O)CCCC3)nn2)cc(C)c(Cl)cc1F c1(C(=O)NC2CCC(CCNC(C3C(=C)C3)=O)C2)cc(F)cc(F)c1OC N1(C(C)C)N=C(C(=O)NCC(C)N(C)C(C2(C)CC3CCC2C3)=O)CCC1=O c1(C(=O)NCC=CCNC(=O)COCCF)cn(CC2CCCOC2)nn1 CCC(C)C(CNC(=O)CCC1(NC(c2csc(C)c2)=O)CCC1)CO c1(C(N(CCNC(C(C)(C)N2CCCCC2)=O)C2CC2)=O)ccc(O)c(Cl)c1 Cc1ccc(C(F)(F)F)cc1NC(C1(F)CN(Cc2cncc(Cl)c2)C1)=O Cn1nc(C(=O)NCC2CCCN(C(=O)C(O)Cn3cncn3)C2)cc1O N1(C(C=C(C)Cl)=O)Cc2ccc(CNC(=O)C(c3c(C)n[nH]c3C)C)cc2C1 c1(C(CNC(=O)NCC2C(OC)CCC2)F)ccccc1Br CC1CCN(C(=O)CC23CCCC2C3)CCN1C(=O)Cn1nc(O)ccc1=O O(NC(=O)C(C)(C)C1CCCN1C(=O)CCC1CC(N(C)C)C1)C(C(C)C)C c1(C(N2C(CNC(c3ccc(C#N)cn3)=O)CCC2)=O)n[nH]c2c1COCC2 c1(COC(c2c(OC(C)C)nccc2)=O)nc2ccccc2[nH]1 Cc1cnc(C(N2CCN(C(c3cccc(Cl)c3F)=O)CC2C)=O)cc1Cl CC1=C(F)CN(C(=O)CC2N(C(C3CCC=CCCC3)=O)CCC2(C)C)CC1 C12(C(=O)NC3(CC=C)CCN(C(C4CC4C(F)(F)F)=O)C3)CCC(CC1)C2(C)C c1(CC)cc(C(N2CCC(C)(NC(=O)CCC(C)CN(C)C)C2)=O)cn(C)c1=O C1(C(=O)NCC2(CC(C)C)CCC2)(NC(c2cccc(C(N)=O)c2)=O)CCN(C)C1 N1(C(CC(C)(C)C#N)=O)CCC2(CCOC2)C(CNC(=O)CSC(=N)N)C1 C1(C(N2CCC(C(CC)C)CC2)=O)C2CC(O)C(C2)N1C(c1cnc(C)o1)=O Cc1nc2c(NC(C3(C)CCCN3C(c3ccc(Cl)cc3C)=O)=O)cccc2s1 c1(CCC(N2CC(NC(c3cc(Cl)cnn3)=O)C3C2C3)=O)cccc(F)c1F C(=O)(C#CC1CCCOC1)N(CC(CNC(c1cc(S(=O)(=O)NC)oc1)=O)C)C CC(CC(=O)N1CC(C(N2CC(O)C2)=O)CC1(C)C)C(F)(F)F c1(C(=O)NC(CC)CN(C)C(C2C=CCCC2)=O)ccc(OC)c(F)c1 c1(OC)ncccc1CC(=O)N(C)CCN(C(=O)CC(C)c1ccncc1)C c1(C(=O)NCC2CCC(NC(C3(Cl)CC34CCC4)=O)CC2)cncc2ccccc12 C1(NC(c2nncs2)=O)CC2CN(C(=O)CNC(c3ccco3)=O)CC12 c1(C(=O)NCCNC(C2CC(C#C)(O)C2)=O)cc(OC(F)(F)F)cc(Cl)c1 N#CC1(CN2C(=O)CN(CC34CCCCC3C4)C2=O)CCCCC1 c1(C(NC2CCN(C(=O)CS)C2)=O)cn(C(F)F)cn1.C(C)(C)SC S(=O)(=O)(c1cccnc1)N1C(C(=O)NC2CCC(F)(F)CC2)CC1 C1(CC(=O)NC2(CO)CN(C(C3(CC)CCCC3)=O)C2)CCC(C)(C)C1 Cn1ccc(C=CC(=O)NCC2(CNC(=O)Cc3cscn3)CC(F)(F)C2)c1 CCCCC(CC)C(=O)NC1COCC1CNC(C1CCC(N(C)C)C1)=O c1(CC)ccc(C(=O)NC2CN(C(=O)Cc3ccnc(Br)c3)CC2C#N)cc1Br c1(C(C)=O)c[nH]nc1C(=O)NCCOCCNC(c1cc(C)ns1)=O N1(C(C(CC#C)NC(c2ccc(C#N)s2)=O)=O)CC(F)(C2CC2)C1 C1(CC(=O)NCC(C)N(C)C(c2cc(Cl)c[nH]2)=O)CCCC(O)C1 c1(C(N2CCCC(NC(C3CC(=O)N(CC4CC4)C3)=O)C2)=O)cc(F)cc(Cl)c1 C(C)(C)(C(F)(F)F)OCC(=O)NC(C)CCNC(C1(F)CCCC1)=O N#Cc1ccccc1NC(=O)CCNC1CCC(c2ccccc2F)C1 C1(C(=O)NC(CN2CCN(C(C3(C(C)C)CC3)=O)CC2)C)CC2(CCCC2)CO1 C1(C(=O)NCC(CNC(C(CSC)O)=O)(C)O)CC2CCCC(C1)C2 C1(NC(C2CCCN(S(=O)(=O)C(F)F)C2)=O)CN(C(c2cnc(Cl)s2)=O)CC1O c1(NC(C2C(C)C3CCC2C3)=O)ccc2c(c1)S(=O)(=O)NC(=O)N2 C1(C(=O)NC2CCCCC2O)CCCCC1NC(CNC(=O)CC1C=CCCC1)=O C(=O)(CCCC(F)F)NCC1CCC(NC(Cc2c(C)nc(CCCC)s2)=O)C1 c1(OCC)ccc(=NC(=O)c2cc(-c3ccc(C)cc3Br)cn3ccnc23)[nH]n1 N1(C(C(CC)C)=O)CC2CN(C(C3(c4ccc(C)c(Cl)c4)CC3)=O)CC2C1 N1(C(C2(COC)CCNC2)=O)CCC(O)(C(F)(F)C(N)=O)C1 C(CC(O)CC(=O)NCCC1CSCCN1C(c1ccc(F)c(C)c1)=O)SC N1(C(c2ccc(C)cc2Cl)=O)CC2CCN(C(c3cc4n(n3)CCO4)=O)C2C1 C1(C(=O)NC(C2CSC2)C)CNC(=O)CN1C(c1csc(Cl)c1)=O c1(CCC)occc1C(=O)N(CCC(=O)NC1CCOC1=O)C1CC1 C1(CC(=O)NC2CC(OC)C2(C)C)CCOCC1(C)C C1(CNC(C(CCC)NC(C)=O)=O)CN(C(=O)CC2CC(F)(F)C2)CC(C)(C)O1 C1(CN2C(C(c3ccccc3)O)CCC2)CC2CC1CO2 N1(C(C2N(CC)CC2)=O)CCCCC(C(=O)N(CC(=O)OC)CC2CC2)C1 C=CC1CN(C(=O)C(F)(F)CC)CC1NC(C1(CC2CC2)CC1)=O CCCC(C)(C)C(=O)N1CC(CC(=O)NCC(C)OCCO)C2(CC2)C1 C1(C(N2C(c3ccc(OC)cc3)CCC(C)C2)=O)CCn2c(cnc2C)C1 C1(CNC(C2ON=C(C)C2)=O)(CO)CC12CCN(C(c1coc(C)n1)=O)CC2 C(C(C(C)(C)C)NC(c1ccccc1C(C)O)=O)NC(c1cn(CCC)nn1)=O N1(C(CCCCCC)=O)CC2CC(NC(=O)CCC(C)O)CC2C1 c1(C(=O)NCC(C)N(C(=O)CCc2cnco2)C)cc(CO)n(C)n1 c1(N2C(CN(C(=O)COCC(F)(F)F)C)CCCC2)ccn2c(Br)cnc2n1 N1(C(C(C)OCOC)=O)CCC(C)(C)C1CNC(=O)Cn1cc(C(F)(F)F)nn1 C1(CNC(CNC(C)=O)=O)CCCC2(CN(C(c3cnc(F)c(C)c3)=O)C2)O1 C(=O)(C(C)(C)NC(=O)C(C)(C)C)NC(CC)CNC(=O)C(C)O c1(NC2(CNC(C(C)SC(F)(F)F)=O)CCCC2)ccc(S(C)(=O)=O)cn1 C1(C(N2CC(NC(C3CC34CC(C)(C)C4)=O)C(C)C2)=O)(OC)CCS(=O)(=O)C1 c1(N2CC(O)(CCNC(C3(O)CCCC(C)(C)C3)=O)C2)nc(Cl)nc2c1CCC2 N1(C(CCC2CC(OC)C2)=O)CCC(NC(c2ncccc2C)=O)C(F)(F)CC1 C1(CCC(=O)NCCn2cc(Cn3c(C)ncc3)nn2)CC(C)(C)CO1 N1(C(C(C)OCC#C)=O)CC2CCCC(C(=O)Nc3cccc([N+](=O)[O-])c3)C2C1 c1(C(C)C)ccc(C(=O)NCC(C)(C2CC2)NC(c2csc(Cl)n2)=O)cn1 N1(C(Cc2c(C)cco2)=O)CCN(C(C2CC2C(=O)OC)=O)C(CF)C1 N1(C(c2ncn(C)c2)=O)CC(C2CCCN(C(=O)C(C)(C)C(F)(F)F)C2)C1 c1(C(C)C)ccc2c(c1)CCC2NC(=O)NC1CCN(Cc2ccccc2)CC1C N1(C(C(C)OC2CCCOC2)=O)CCC2(CCCCC2NC(=O)COC(F)F)C1 Cn1cc(Cl)c(C(=O)NCCCCCCNC(C2(C)CCCOC2)=O)n1 c1(C(=O)NC2CN(C(=O)OCC)CC2C)cc(NC(c2cnco2)=O)n(C)n1 CC1(C)COC(CC(N2CC3C(NC(=O)Cn4ccccc4=O)C3C2)=O)CO1 CC1(C)C2CN(C(c3onc4ccccc34)=O)C(C(=O)NCC3(O)CC3)C12 c1(C(=O)NC2(C)CCN(c3c(OC)cncn3)CC2)ccc2cncn2c1C c1(CC(=O)NCCNC(C23OCC(COC)(C2)C3)=O)ccccc1S(C)(=O)=O N1(C(C(=O)NC)=O)CCOC2(CCS(=O)(=NC(=O)C3CC4CC3C3CC43)CC2)C1 c1(N(C2CCCOC2)CC)ncc(C)cc1Br c1(C(=O)NC(CC)CNC(=O)C(F)Cc2ccccc2)c(S(N)(=O)=O)cnn1C c1(C(=O)NCC(C)CNC(C2CCCN2C=O)=O)cnncc1O c1(NC(C(C)NC(=O)NC23CC(C2)C3)=O)ccc(Br)cc1Cl C1(CS(=O)(=O)NC(c2cccc(C)c2)C)CC(C)(C)OC1(C)C N1(C(CCn2c(C)nc([N+](=O)[O-])c2)=O)CC2CC(C1)CN(C(c1cocn1)=O)C2 C(=O)(C(C)C(C)c1ccccc1)NC(C(=O)OC)CN1CCCCC1 c1(C(=O)OCC)cccnc1NCC1CCC(NC(=O)C(c2ccncc2)C)C1 C#CC1(O)CC(C(=O)NCC2(NC(C3CC34CC4)=O)CCOCC2)C1 C(C(O)(CNC(=O)C(CCF)NC(=O)CC=C(C)C)CO)OC C(=O)(C(O)C(C)(C)C)N(C(C)C(=O)NCc1cnc[nH]1)CC c1(C(N2CC(CC)C(NC(=O)CC(C)CF)C2)=O)ccc2nc(N(C)C)sc2c1 CC1CCN(C(c2cccs2)=O)C1C(=O)NCC1(C#N)CCCC1 c1(CN2CC3C(NC(=O)CC4CC4)C3C2)ccc2c(c1)CCC2 O=C(CC1CCCN1C(c1n[nH]c2cccnc12)=O)N=c1ccnc(Br)[nH]1 c1(CC(=O)Nc2ccc(F)cc2)cncc(C2CC2)n1 C1(NC(CC(C)n2cccn2)=O)CN(C(c2cc(C3CC3)on2)=O)CC1C C(C)(N=c1ccc2c([nH]1)CCCC2=O)c1c(NC(C(C(C)C)OC)=O)cccc1 C(c1ccc(S(=O)(=O)NC23CCC(CC2N)C3)cc1)=CC(=O)NC1CC1 c1(CCC(=O)NC(CNC(CC(=O)NCC#C)=O)C(C)C)ccccc1C(N)=O N(C(=NCC(C)C)NCC12CCC(C)(CC1)CO2)Cc1cc(CC)[nH]n1 N1(C(C23OCC(COC)(C2)C3)=O)CC2CC(C1)C2NC(=O)C(c1ccccc1)O O=C(CC(C(F)(F)F)n1cccn1)N1CCC(CNC(C2(CCF)CCC2)=O)C1 C1(C(C)=O)CCCN(C(=O)NC2(c3cn(CCC4CCCO4)nn3)CC2)C1 C1(NC(C2N(C(CC3CC(C)C3)=O)CC(C)C2)=O)CNC(=O)C12CC2 C(CC(=O)NC1(C(=O)NC(c2cncs2)C)CC1C)SCC c1(SC)nccc(N2CCCCC2C(=O)NCCSCc2ccccc2)n1 c1(C(=O)NC2C(NC(c3c(F)cc(OC)cc3F)=O)C2)cc([N+](=O)[O-])ccc1C c1(C(N2C(CNC(CC(C)OC)=O)CC(O)C2)=O)ccc2c(c1)C(=O)OC2(C)C C12(C(=O)NC3CC4C(NC(c5ccc(COC)cc5)=O)C4C3)CCCC1OCC2 Cc1nc(C2CC2)[nH]c1C(=O)NCCCC1CCCN1C(c1n[nH]cc1Cl)=O C=CCC(CC(F)F)C(=O)NC1C2CCN(C(C3C(C)(C)C3(F)F)=O)CC12 CC12CN(C(=O)CCc3cccc(Cl)c3)CC1CN(C(=O)C(O)P(C)(C)=O)C2 N1(C(C(C#C)(C)C)=O)C2CCC1CC(CCNC(=O)CCNC(C)=O)C2 Cc1cc(Cl)c(C(=O)CNCC(O)COc2ccc(CC(=O)NC)cc2)cc1C c1(CC(=O)NCC2C(C)(C)N(C(C3CC=CCO3)=O)CC2)cc(F)c(F)cc1F c1(OC)ncc(Br)cc1CN1CC(C)CC1C(=O)NCC1CCO1 C(=O)(CCCCC(=O)NCC1(CCNC(c2ccnc(C)c2Cl)=O)CC1)OC N1(C(CC2CC(C(=O)OC)C2)=O)CC2CC(C1)N(C(C1OCCC1C(C)C)=O)C2 C1(CC(=O)NC(C(=O)NCC(CC(C)C)NC(N)=O)C)CN2CCN1CC2 N1(CCC)CCCCC1C(=O)NCC1COCCN1C(=O)C=CC(=O)OCC C12(C(=O)NCC3N(C(c4cc(CC)on4)=O)CC3)CC3CCC(CC(C3)C1)C2 CC(C)C(C)(CNC(c1ccncc1O)=O)NC(=O)CCC1CCC1 c1(C(=O)NC(C(c2ccccc2)NC(CC(C)O)=O)C)ccc2cc[nH]c2n1 N#Cc1ccc(C(N2CCCC2C2(NC(=O)CC3CCC(=O)N3)CC2)=O)nc1 C1(C(=O)NC(C(=O)N2CC(c3c(C)con3)C2)CC2CCCC2)CCCCC1F C1(N(CCNC(N2C(C(C)O)CC2)=O)CCO)CCCCC1 C(=O)(N1CCC(C(=O)NC2C3CCCCCC23)O1)C1(N(C)C)CCC1 c1(C(N2C(CNC(=O)CSc3ncccn3)CCC2)=O)cnc2c(c1)CCOC2 c1(C(=O)NCCCC(C)NC(C2(Cl)CC2)=O)cncc(-c2ccccn2)c1 N1(CC)CCCCC1C(=O)NCC1CCCC1NC(=O)CCCOC C(CCCCC(=O)NCCC1CC(NC(c2nocc2C2CC2)=O)C1)OC C1(c2n(CC=C)nnn2)(Nc2cccnc2C)COC2(CCOCC2)C1 c1(SCC(=O)NCCC2(NC(=O)NC3C4COCC34)CC2)ccccc1 C12(CCCSC1)C(=O)N2.c1(C(C)(C)C)[nH]cnc1C(=O)N(C)CC1C2COCC12 N1(C(c2cn(CCNC(C(CC)SC)=O)nc2)=O)CC(O)C(O)C1C(=O)O N1(C(C2(C=C)CCCC2)=O)CCCC(F)(CNC(C2CC(=O)N(O)C2)=O)C1 Cc1ccc(SCC(N2CCOC(CCCNC(C3CC(C)(O)C3)=O)C2)=O)cc1 C1(NC(CCC(=O)NCCC)=O)CN(C(=O)Cc2nonc2C)C(C)(C)C1 C(=O)(CC(O)C1CCCC1)NCC(=CC(=O)N(C(CC)C1CC1)C)C C(=O)(C(O)(C(C)C)C(F)(F)F)NC1CN(C(c2cc(OC)ns2)=O)CC1C C12(CC(=O)N(C3CCN(C(=O)CCS(N)(=O)=O)C3)C)CCCN1CCC2 C1(NC(CCC(C)OC)=O)CC2(C1)CC(C(=O)NC(C)C(=O)OC(C)C)C2 CC(N)CCC(=O)N1CCOC(CCc2ccccc2)C1 c1(C(=O)NC2CC(CCNC(Cn3c(C)ncc3)=O)C2)cc(N(C)C)ccc1N C(=O)(C(S(C)(=O)=O)C1CC1)N1C(CNC(C(C(C)C)NC(=O)OC)=O)CC1 N1(C(C(CC(=C)C)C)=O)CC2CCOC2(CNC(c2cc(N)ccc2C)=O)C1 c1(NC(C23C(C)OC(C)(C2)C3)=O)ccc2nccnc2n1 c1(OCC=C)ccc(CC(N2CC3CC3(CNC(C3CC(CF)C3)=O)C2)=O)cc1 c1(NC(C2N(c3nc(OC)cc(OC)n3)CC3(CC3)C2)=O)cccc(C#N)c1Cl N1(C(c2cc(CC)cc(N)c2)=O)CC2CCC(C1)C(NC(C1CC1F)=O)C2 c1(C(=O)OCC)cc(=NCCCOCC(=O)OCc2cc(C)oc2C)[nH]c(C)n1 CC1(C(=O)NCCOCCNC(=O)Cn2cc(C(C)O)nn2)CNC(=O)C1 C1(C)(C(=O)NC(CC)(C)COC)CCN(C(=O)C2=CCOCC2)CC1 N(C1COc2cc(Br)ccc21)C(c1nnc(C)n1C)C(=O)NC1CCOC1 N1(C(c2c(C)nn(C(C)C)c2C)=O)CC2CN(C(c3cc(Br)c[nH]3)=O)CC2C1 c1(NC(C)=O)ccc(N)c(C(N2CC(F)(F)CC2CCNC(=O)CC(C)C)=O)c1 C#Cc1ccc(C(=O)NCCC(C)NC(=O)C(C)(O)C2CCC2)nc1 C(CCC(O)CO)N(C)C(C1CC(C)(NC(=O)CC2OCCCO2)C1)=O CCC(CC)(CC)C(=O)NCC12CC1CN(C(=O)Cn1cnc(C(N)=O)n1)C2 C1(C(N2CCC(NC(c3c(CC)scn3)=O)(CF)C2)=O)(CC)CCC(O)CC1 C1(C(=O)NCC(C)CN(C)C(C2CC23CC3)=O)CCC2(CC1)NC(=O)N(C)C2=O c1(OC)cc(C(=O)NCCCOCCNC(C2CCS(=O)CC2)=O)nn1C CC1(C)CCC=C(C(=O)NC2CN(C(=O)CCc3cnc(O)[nH]3)CC2C2CC2)C1 Cc1cnc(Cl)nc1N(CC(C)NC(c1ccc(-c2cc[nH]n2)s1)=O)C c1(C(=O)NC2COC3(C2)CN(C(=O)CCC2CC2)C3)cc2ccncc2c(O)n1 C1(N(C(c2c(C)scn2)=O)C)CCCN(C(c2cc[nH]c2-c2ccccc2)=O)C1 c1(C(=O)NCC(N(C(C2N(CCC)CCC2)=O)C)C2CC2)c(F)cc(F)cc1Cl c1(C(=O)Nc2nc(C)c(I)s2)csc2c1CCN(C(c1cnc(Cl)cc1I)=O)C2 C(=O)(C1CCCn2cnnc21)N1CCN(C(C(CCCCC)(C)C)=O)CC1C c1(OC)ccc2nc(CNCC34CC=CC(C3)OC4)ccc2c1O N1(C(C=C(CC)CC)=O)CCCC(N(C(=O)CCSC)CC)CC1 c1(C(=O)NC(CCOC)CNC(c2nn(C)cc2C)=O)ccc(N=[N+]=[N-])cc1 N1(C(c2cc(OCC)n[nH]2)=O)CCC(O)C(C(=O)NCC2CCCO2)C1 c1(NC(C2CCCC2NCc2ccc(Br)cn2)=O)cccc(O)c1Cl C1(F)(C(N(CCCOC(C)C)C)=O)CCN(C(=O)C(C)O)C1 c1(C(=O)NC(CNC(C)=O)C(N)=O)nnn(-c2ccccc2Cl)c1C c1(C(=O)NC2CC(NC(C(CCC)O)=O)CC2O)cc2c(nn1)OCCS2 c1(NC(C(=O)NCc2n(C)ncn2)=O)ccc(F)c(N2C(=O)CNC2=O)c1 C1(OCCC)CCCCC1C(=O)NC(C)CNC(c1cccc(N(C)C)n1)=O C1(F)(C(=O)NCC2(NC(c3n(CCC)ncc3)=O)CCC2)C2CCCC12 c1(CC(C)NC(C2(c3cccc(C)c3C)CCCC2)=O)c[nH]c2c(C)cccc12 c1(C(=O)NCC2C(CNC(c3csc(C(F)F)n3)=O)C2)c[nH]c2cccc(F)c12 c1(CNCC(C)(O)c2cccs2)cc(Br)cc(Cl)c1F N1(C(C(C)(O)C2CCC2)=O)CCOC(CCNC(c2nocc2Br)=O)C1 CCC(c1ccccc1)=CC(=O)NCC(O)CN(C(=O)CC1CC1)C C12(CC)COC(C(=O)Oc3ccsc3Cl)(C1)C2.C12CCN(CC1)C(=O)CS2 c1(C(N2CC(F)(CNC(CCC3C(C)C3)=O)C2)=O)ccc(Cl)c(N)c1Cl c1(C(N2CC(CC=C)(NC(=O)CCC(=C)C)C2)=O)cn(C)c2ccccc12 c1(CN2C(C(=O)Nc3cn(C)nn3)CC2)ccc(C#N)c(Cl)c1 C1(C(N(CCNC(c2cc(O)ccc2Cl)=O)CC2CC2)=O)CC2CCC1CC2 c1(N2C3CC(CNC(C4CCC(C)O4)=O)CC2CC3)ncccc1S(C)(=O)=O CC(C(=O)NC1(CO)CCN(C(c2ccccc2CO)=O)CC1)C(C)(C)O c1(N(CCn2c(C)ncc2)C)nc2c(c(=NCCC3CC3)[nH]1)SCC2 c1(OC)ccc(C(=O)NC2(CNC(C3CCC(F)(F)C3)=O)CCC2)c(C)c1OC CCN=c1[nH]c(C(=O)N(C2CCCCN(C(=O)CCNC(N)=O)C2)C)cs1 N1(C(c2cc(C)c(Cl)s2)=O)CCCC12CCCN(C(=O)CCc1cnn[nH]1)C2 C1(C(=O)NC2CCN(C(=O)OC(C)(C)C)C2)COCCN1C(=O)CCC(N)=O CC#CCC(C(=O)NCCC(C)C(F)(F)F)NC(=O)CCOC n1(C(C)C)nnnc1C(C1CCCCS1)NCCc1ccccn1 C(C(C)(C)C(c1nnnn1C1(C)CC1)Nc1ccc(SC)cc1)(OC)OC C1(C(N(CCCC(C)NC(C=CCC)=O)C2CC2)=O)CCC(C(C)C)NC1=O N1(C(COC2(C)CCOCC2)=O)CC2CCC1C(CN=c1[nH]c(Cl)ncc1Br)C2 N1(C(C2CCCN(C(=O)OC)C2)=O)CC2CCC1C2NC(C1CCC2CC12)=O c1(-n2ncc(C)c2)ccnc(NC(C2CCN(c3ccccc3Cl)C2)=O)n1 C1(C(C)(C)NC(=O)CCc2ccon2)CCN(C(c2cc(Br)c[nH]2)=O)C1 C1(O)(C(N(CC=C)C)=O)CCOC1(C)C.N1CCCC(ONC(=O)C=C(C)C)C1 c1(C(N2CC(NC(c3ccoc3Br)=O)(CO)C2)=O)ccnc2cc(F)cnc12 C(C)(CNC(=O)CN1CCN(S(C)(=O)=O)CC1)(CC(C)C)NC(C(CSC)O)=O Oc1cc(-c2ccc(-c3ncc[nH]3)cc2)c2ccccc2n1 c1(CCC)cccc(C(=O)N(C)CCNC(c2cn(C(F)F)cn2)=O)c1 C(=O)(C(C)(C)C1CCOC1)NCC(C)(C)OCC(=O)Nc1cnn(C(F)F)c1 c1(C(=O)NCCCC(C)(C)NC(=O)C(CO)C(C)(C)C)ccc([N+](=O)[O-])cc1 CCC(C(C)(C)O)NC(=O)CCN(CCCO)C(C1CCC(CSC)CC1)=O N1(C(c2ccc(OCF)cc2)=O)CCN(C(=O)C(O)Cn2cncn2)CC1CO CC1(C)C(C(=O)NOCC(=O)NCCOC2CC2)C1(C)C C1(CNC(C2(C)CCNC2=O)=O)CC2CC1CN2C(c1cncc(N)n1)=O C(=O)(C(C)CC(N)=O)NC1CC(NC(c2c(COC)ccs2)=O)C1 C1(NS(N(C2CCNCC2)CC)(=O)=O)(CC)CC2CCC1CC2 C1(NC(CCN(C(=O)CNC(=O)NC)CC=C)=O)CCCC1C CCC(C)(O)C(=O)NC1CCCC1C(=O)NC12CCCC1C2 C=CC1(C(=O)NC(Cc2ccco2)CO)CCN(C(=O)C(F)C(=O)OCC)C1 C1(C(=O)NCCCn2cc(CCCSC)nn2)CCC2CCCC2O1 c1(CC(N2C3CCC(NC(CN(C(C)=O)C)=O)C(C3)C2)=O)ccc2c[nH]nc2c1 CC1CCC(O)(C(N2CCC(C(C)C(=O)NCCc3nccs3)C2)=O)CC1 C1(COC)(NC(=O)CCc2ccsc2)CCN(C(=O)CC2(C(F)(F)F)CC2)CC1 C1(C(=O)NC2CCN(C(c3cnc(SC)n3C)=O)C2)CCn2ncnc2C1 C12(C(=O)NCCC(CNC(c3c(CC)nccc3)=O)O)CCC(C1)OC2C C1(N=c2[nH]ccnc2F)(CCC)CCN(C(=O)C=Cc2ccnn2CC)CC1 c1(OC)ccc2[nH]c(C(N3CC4CN(C(=O)C(N)=O)CC4(C)C3)=O)cc2c1OC CC1CN(C(=O)C(N)=O)CC2(CCN(C(=O)COCCCN(C)C)C2)O1 C(C(F)(F)CCC(=O)Nc1c(C)nsc1C)SC N1(C(C2C(CC)OCCC2)=O)CC2CN(C(c3ccc(F)c(OC)c3)=O)CC2C1 N1(C(Cc2n[nH]c(=NC)s2)=O)CCN(C(=O)C(C2CCC(=O)N2)C)C2(CC2)C1 c1(OCCOC)ccc(C(=O)N(C(C)CNC(=O)Cc2cnc[nH]2)C)cc1 C(=O)(C1c2c[nH]nc2CCC1C)N1CC2CC(CN(C(CC(C=C)(C)C)=O)C2)C1 N1(C(C(CC)N(C(=O)Cn2nnn(CC)c2=O)CC)=O)CCC(C)C1(C)C C1(OC)CCCCC1NC(C1OCCC1NC(=O)C(CN(C)C)N(C)C)=O N1(C(CCC(C)SC)=O)CCN(C(c2cn(C)c(O)n2)=O)C(C2CCC2)C1 N1(C(=O)CC2COCC2O)CCOC2(C1)CN(C(=O)Cc1ccns1)C2 C1(OC)CC2CC(C1)N(C(C1CCCN(C(=O)CC34CCCN3CCC4)C1)=O)C2 C(=O)(C(CCCC(OC)OC)NC1CCCCN1C(=O)OC(C)(C)C)NCC c12cc(nc(SC)n1)S2.C(=O)(C(O)C(C)C)N1CCC(CCC)C1 c1(CC(C(=O)NC(C)C)NC(c2nccs2)CC2CC2)cccc(Cl)c1 c1(C(N2CCC(CN(C)C(C3(Cl)CC34CCC4)=O)C2)=O)cc2ccccc2s1 N1(CC(=O)OCC2CCOC2)CCOCN1c1ccccc1 c1(C(=O)NC2CC2NC(C2CC(Cl)(Cl)C2)=O)cc2c(F)cc(Cl)cc2[nH]1 C(=O)(CC(C(F)F)NC(=O)C(O)C(F)(F)F)N1CC2C(CC)(C2)C1 c1(C(N2CCC(NC(c3cc(C)n(C)c3)=O)C(C)C2)=O)cccc2c1CCCC2 CC12CCC(C(=O)NC3CC4(C3)CC4NC(c3cnc(C(F)F)s3)=O)(CC1)CO2 CC1(Nc2ncc(C(F)(F)F)cc2Cl)CCC(NC(C2CC23CCCC3)=O)CC1 CC(CC(=O)NC1CCCC1CNC(c1cnco1)=O)C(C)(C)C Cc1cc(Br)ccc1CN1CCC(C(=O)NCc2ccccn2)C(O)C1 OC(CN=c1ccc2c([nH]1)OCC2)C1CCNCC1 CC(C)(CC(=O)N1CCC(C(F)CNC(=O)CSC2CC2)CC1)C1CC1 C(=O)(C1Cc2ccccc21)N1CCC2(C(C(=O)NC(C(CC)C)CO)C2)CC1 C1(C(N2CC(O)(C(C)NC(c3ccc(CC)o3)=O)C2)=O)CC2(CC2)CO1 CCC(C)C(C(=O)NC1CC(F)(F)C1)NCC1(c2cccs2)CC1 C1(CCNC(C2CC3CC2C3)=O)CSCCN1C(=O)Cn1cc(C(F)(F)F)cn1 Cc1ccc(F)c(C(N2CCC(O)C(C(N3CC(O)C(F)C3)=O)C2)=O)c1Br c1(C(N2CCOCC(CNC(c3cncc(F)n3)=O)C2)=O)cc2ccccc2o1 C(CNC(c1ccc(C2CC2C)o1)=O)(CC(C)C)NC(CCc1cnc(C)s1)=O Cc1ccc2nc(Cl)c(CN3CCCC3C(=O)Nc3ccc(F)nc3C)cc2c1 C1(C(N2CC(n3cc(-c4cn(CC)nc4)nn3)C2)=O)(OC)CCC(C)C1 c1(CC)cc(NC(=O)C=CCN(C(=O)CC2OCCC2(C)C)C)cnc1C N1(C(=O)CCCc2cccs2)CCC2CN(C(C3CCC(C(F)F)CC3)=O)CC12 C(=O)(CCP(C)(C)=O)N1C(CCNC(=O)CC2CCC(=O)O2)CC(OC)C1 N1(C(CCCNC(=O)OCC)=O)CC2CN(C(=O)CC3CCCC3)CC2(C)C1 N1(C(C(COC)COC)=O)C2CCCC1CC(NC(c1cnccc1F)=O)C2 N1(C(C2OCCN(C)C2)=O)CCCC(O)(CNC(c2ocnc2C(F)F)=O)C1 N1(C(C(C)NC(c2ccco2)=O)=O)CC(N(C(=O)C=CC2CC2)C)C(C)(C)C1 C#Cc1ccccc1CC(=O)NC(C)C(C(C)C)NC(=O)C=C(C)Cl C1(O)(C(C(=O)NCC(N)=O)NC(=O)Cn2cc(Cl)cn2)CCCCC1 C1(NC(c2c(CC)n(CC)nc2)=O)CC2CC(C1)N(C(c1cc[nH]n1)=O)C2 C(CCC(C)CC(=O)N1CCC(NC(c2c(C)nc3sccn23)=O)C1)=C(C)C Cc1ccc(F)c(CC(=O)NC(CNC(=O)CC(F)(F)F)CC(F)(F)F)c1 C1(C(=O)NCC2(C(=O)Nc3cncc(Cl)c3)CCCO2)CCCC12CCC2 c1(C(=O)NC2C(NC(CCC3CCCN(C)C3)=O)CC2)c(F)cc(F)cc1F C(CCC)(C(=O)NCC(C(=O)N(C(CO)C(C)C)C)N(C)C)=CCC N1(C(c2cc(C3CCC3)on2)=O)CC2CCN(C(C3SCCCS3)=O)C(C2)C1 N1(C(C)CCO)CCC(C(C)NCC(c2ccccc2)C)CC1 N1(Cc2c(OC)cc(Cl)cc2)CC2CC(NC(C3CC34CCOCC4)=O)CC1C2 Cc1nccc(S(=O)(=O)N2CCCC(C3CCCN3C(=O)OC(C)(C)C)C2)c1Cl Cc1cncc(C(=O)N(C)Cc2ccccc2CNC(=O)COCP(C)(C)=O)c1 c1(C(=O)NCC(CNC(c2cncnc2C)=O)OC)cc2ccccc2c(=O)o1 C1(NC(CCCCC)=O)CCN(C(=O)CC(C)(C)C2CC2)C(C2CC2)C1 N1(C(C(N2C(=O)CCC2=O)C)=O)CCCN(C(=O)Cc2ccc(Cl)cc2)C(C)C1 C1(NC(CC(CC)SC)=O)CC12CCN(C(C1(C)CC3(CCC3)C1)=O)CC2 C1(OC(C(N2CC(CC(C)NC(=O)CN(C)C3CC3)C2)=O)C)CCCCC1 C1(C(=O)OC)CN(C(=O)C(=O)N(CCCSC)C)CC(C)O1 c1(C(=O)NC(C2(O)CN(c3ncnc4sccc34)C2)C)c[nH]c2ncccc12 CC12CCOC(C(N3CCN(CCCNC(C4(Cl)CC45CCC5)=O)CC3)=O)(C1)C2 c1(OC)ccc2cnnc(N(C)C(c3ccc(Cl)cc3)C)c2c1 C1(C(N(C)CC2N(C(c3nccc(C)c3)=O)CCCC2)=O)CCn2cnnc2C1 c1(C(=O)NCC2CN(C(c3c(C)cno3)=O)CC2(F)CO)cc2c([nH]1)CCOC2 c1(C(N2CCOCC2CNC(=O)C(F)(F)CC2CCCO2)=O)ccc(Cl)cc1O C1(CC)CCCN(C(c2cc(O)cs2)=O)C1C(=O)NCC(C)(C)C(C)O c1(C(c2nnnn2C(c2ccccc2)C)NCCOC)c[nH]nc1C C1(CC(=O)NCC(C)(C)CNC(c2occc2F)=O)CCC12CCC2 Cc1ccc(N(C)C(C2OCCC2CNC(C2(O)CCOC2)=O)=O)cc1F Cc1cc(C(=O)NC2CCCC(NC(c3csc(C(N)=O)n3)=O)C2)nn1C1CC1 c1(OC)cnccc1CN1CCC(C(C)NC(C2(CC(C)C)CCC2)=O)CC1 N1(NC(=O)NCC(C)(CN(C)C(c2sccc2C2CC2)=O)OC)CCOC(C)C1 C1(CC(=O)NCCC2C(C)(C)OCC2)C2CCCC2N1C(=O)Cc1csnn1 C(=O)(CC1(CN(C)C)CC1)NC(C1CC1Cl)C N1(CC)CCCC(N(C(=O)C2CC2)NC(c2cn(C)nc2CC(C)C)=O)C1 c1(CC)nnc2c(C(N3CCC3CNC(=O)C(c3cccnc3)O)=O)cccn12 c1(SC)ccccc1C(N1CC(NC(c2c(Cl)cnn2C)=O)C(SC)C1)=O C1(C(=O)NC)CN(C(C2CC2(C)C(F)F)=O)C1 CN1CCCC(F)(C(N2CC(O)(CCNC(=O)CCNS(C)(=O)=O)C2)=O)C1 C(=O)(C1=NOC(C)C1C)NCC(CC)N(C(=O)CCCc1ncco1)C c1(CC)ccc(C(=O)NCC2CCCN2C(=O)C(F)C2CC2)cc1[N+](=O)[O-] N1(C(c2c(CC)ccs2)=O)C2CCC1CC(NC(=O)C(C)(F)C(C)(C)F)C2 C(=O)(C(O)P(C)(C)=O)NCC(C1CC1)NC(c1cn(C)nc1C1CC1)=O CC#CCCCC(=O)N1CCC(O)(C(C)NC(c2cnn(-c3nccs3)c2)=O)C1 C(=O)(C(O)P(C)(C)=O)N1CCC(NC(CC=CC=C)=O)(COC)C1 C1(OCC(=O)NC(C2CCN(C(C3CCC4CC34)=O)C2)C)CCN(C)CC1 C1(NC(C(COC(C)C)NC(c2ccncc2F)=O)=O)CCCC(F)(F)C1 CCC(CC(=O)NCC(CC)CCO)N(C(=O)CCC(=O)N(C)C)C n1(CC(N2CC3C(C(=O)NC4CCNC4=O)C3C2)=O)nc(Cl)ccc1=O C(c1cc(OC)ns1)=CC(=O)N(CCNC(=O)CCc1cc(Cl)no1)CC C(=O)(C1CCc2c[nH]nc21)N1CCN(C(C2=CCC(C)CC2)=O)CC1C(C)(C)C Cc1ccccc1OCc1nc(CN(C(=O)CSc2ccncc2)C2CC2)cs1 C1(O)(CNC(C(C)N(C(=O)COCCCOC)CCC)=O)CC2CCC1O2 N1(CC(=O)NCCC2CN(C(c3cn(C4CC4)cn3)=O)CCO2)CC(=O)NC1=O N1(C(COCCOCC#C)=O)CCCC2C1CCN2C(=O)Cc1c[nH]nc1C S(=O)(=O)(CC(=O)N1CCN(C(=O)CC2COCCN2C)CC1)NC N1(C(C(c2cccc(C)c2)=O)=O)CC2CC1CN(C(=O)CCC1CNC(=O)N1)C2 C(C(CC(C)C)NC(C1CC(n2ccnc2)C1)=O)NC(c1nc(C)oc1)=O CC1(O)CC(C(=O)NCC2CC(C(N3CCCC3CN=[N+]=[N-])=O)CO2)C1 N1(C(=O)C=Cc2nccs2)CCC(=CCNC(C2(n3cncn3)CC2)=O)CC1 N1(C(c2ccc(C)o2)=O)CC2(C(=O)NCCC(F)(F)CO)CCC1CC2 Cc1nc2cncc(C(=O)N(C(C)CNC(C3CCCSC3)=O)C)c2[nH]1 c1(-c2cn(C(C)CNC(c3cnccn3)=O)nn2)ccc(S(C)=O)cc1 C(=O)(C(C)(C)CC1CC1)N1CCC(CN(C(CC2(CSC)CC2)=O)C)C1 N1(C(c2n(CC)nc(C)c2)=O)CCC2(CCCC2NC(=O)CSC(F)F)C1 N1(C(C2(CCN(C)C)CC2)=O)CC2(C(N3CC(CO)CC3CO)=O)CCC1CC2 N1(C(CC2CC(=C)C2)=O)CC2(CCN(C(c3ccc(CC(C)C)nc3)=O)C2)C1 c1(C(=O)OCC)cnn2c(C(=O)N(CCCNC(C)=O)C)ccnc12 Cc1ccc(CCNC(C2(O)CCN(C(=O)CS(C)(=O)=O)C2)=O)cc1 CN1CCCN(C2CCN(C3CCCN(C(=O)COCC(=O)O)CC3)CC2)CC1 N1(C(=O)Nc2ccc(OC(C)C)c(Cl)c2)CC2C(C(F)(F)F)(C1)CS2(=O)=O C1(C(N2CC(C)(CCC(=O)NC(C(C)F)C)C2)=O)C2CCC(C2)C1C C1(CN(C(C2C(OCC)C2)=O)C)CCC(NC(C23CC(F)C2C3)=O)CC1 C1(NC(=O)COCCF)CN(C(=O)Cc2cc(F)ncc2Br)CC2(CC2)C1 c1(C(N2CCC(NC(C(CCOC)C)=O)CC2)=O)c(Br)c(C)nn1C CCCC(C(=O)OC)C(=O)N1CCC(C2CC2)(NC(C2CN(C)C2)=O)C1 N1(C(C(C)N(C)C(C2CC3C(C2)C3(F)F)=O)=O)CCC2(CCOC2=O)C1 c1(C(=O)NCC2(F)CC(NC(C3(CCF)CCC3)=O)C2)c(F)cc(Cl)cc1F N1(C(c2ccc(C(C)C)o2)=O)CC2CC2(C(=O)NCCCC2CC2)C1 Cc1cc(C(=O)NCC2(O)CN(C(=O)Cc3cnn(C4CC4)c3)C2)cc(N)c1Cl C(c1ccccc1)=CCN1CCC(CC(=O)NCCC2CC2(Cl)Cl)C1 c1(C(=O)NCCCOCCN(C(CC(CC)C2CCC2)=O)C)ncc(C)cc1F C1(CNC(C(Cn2cncn2)NC(CNC(C)=O)=O)=O)CCC(O)CC1 C(=O)(C1CCCc2ncnn21)NC1(CNC(CC(=O)Nc2nccs2)=O)CCC1 CCC(CC(=O)NC1(COC)CN(C(c2nnn(C)c2C(F)F)=O)C1)SC C(=O)(C1=CCCCO1)N1CCC(NC(c2c(CC)ccs2)=O)(CO)C1 c1(-n2cc(CCCOC(=N)O)nn2)ccc(C)c(C#N)c1.CCC1(C)CNC1=O c1(NCC(C(C)(C)C)NC(CC(C)C)=O)cc2nn[nH]c2cc1[N+](=O)[O-] CC(C)CC(CNC(c1csc(CN(C)C)n1)=O)NC(C1CCC(C)C1)=O C1(C(=O)NC(c2cnc(C)s2)C)CC2(CCN1C(=O)C=CCN1CCCC1)CC2 C(c1cncn1C)=CC(N1C(CNC(C=C2CCC(C)C2)=O)C=CC1)=O C(CC)(CC)(CCNC(=O)C(C)(C)C(C)C)NC(C1(CC#C)CCCCO1)=O C1(C(N2CC3(CNC(C4(CO)CCCO4)=O)CC2CO3)=O)CC2CCCCN2C1 Cc1c(C(=O)NC2CN(C(C3CCCN3C3CCCC3)=O)C2)cncc1Cl C1(CC)CCC(C)N(C(c2oc(CNC(=O)CCCC3CCCC3)cc2C)=O)C1 Cc1ccc(CN2CCCC(C(N3CCCCC3CO)=O)C2)c([N+](=O)[O-])c1 C1(NC(COCCCCCC)=O)CCC(C)(CNC(C2(C)CCCOC2)=O)CC1 C12(C(N(CC)Cc3ccccc3)=O)CC1CN(C(c1ccccc1SC)=O)C2 CCC(C)CC(C)N(C)C(=O)Nc1cn(Cc2ccco2)nc1C1CC1 C(C1=CCN(C(C2CC(S(C)(=O)=O)C2)=O)CC1)NC(c1on(C)c(=O)c1)=O C(=O)(C#CC1(C)COC1)NC1CCCC(NC(c2nn(C)c(C(F)(F)F)c2)=O)C1 Cc1cc(C(=O)NCC2CC(O)CN2C(c2csc(C)c2)=O)cc(O)c1 Cc1nn(C)cc1C(=O)NCC1CCCC1NC(=O)C(c1cn(C)nc1C)C Cc1nc(C)c(CCC(=O)NCC(C)NC(c2c(C)nnn2C)=O)c(O)n1 O=S(=O)(c1ccc(Br)s1)NCc1ccc(Cl)cc1.c1(C2C(=O)N2)cnn(CC)c1 N1(C(C=CC)=O)CCC(C(=O)NCC=CC=Cc2conc2C(C)C)C1 N1(C(c2ccc3nnnn3c2)=O)CCCCC1C1CCCN1Cc1cocn1 C=CC(CCC)CC(=O)N(CC(=O)NCc1ccccc1O)CCC c1(C(C=C=C)C)nc(-c2cncs2)nn1CC c1(C(=O)O)cccc2c(C(=O)NC3CCN4CCCCC34)cccc12 Nc1cc(C(=O)NC2CC(F)(CNC(c3cc4cscc4s3)=O)C2)ncc1Cl CCCCC(O)CC(=O)NCCCC(C)(C)NC(C1CCCCC1C(=O)OC)=O C(=O)(C(C)S(=O)(=O)C(C)C)NC1CC2N(C(CC(=O)NCC#C)=O)C(CC2)C1 N1(C(C2(SC(C)C)CC2)=O)CCC2CCCC12C(=O)NCC(C1CCCC1)OC c1(C(=O)NCCNC(C)C(=O)Nc2ccc(OC(F)(F)F)cc2)cn(C)nc1Cl C(=O)(C1CCc2c[nH]nc21)NCC(C)CN(C(=O)CCSCc1ccccc1)C C1(N(c2nscc2NC(c2ccccn2)=O)C)CCCN(Cc2cnn(C)c2)C1 C1(NC(c2c(OCCC)cccc2)=O)CCN(C(=O)CCOC(C)=O)CCC1CO CC(C)C(C(=O)NC(C1CN(C(c2nc(C3CC3)cs2)=O)C1)C)c1cnn(C)c1 c1(CNC2C(C(=O)Nc3ccc(O)nc3)C2)c[nH]c2ncc(Br)nc12 S(=O)(=O)(c1cc(OC)cc(F)c1)NCC(C)C#N c1(CNC(C(N2CCC(O)(C(=O)OC)CC2)=O)=O)cc2c(cc1O)OCO2 CC1CCCC(OCC(N2CCOC(CNC(=O)C(F)=CCCF)C2)=O)C1 C1(CC(=O)N(C2CCCOC2)CC)CCC(NC(=O)CCOC(C)=O)C1 C1(CNC(=O)CC2CCC3CC3C2)COCCN(C(C2(O)CCOC2)=O)C1 C(CCN=c1ccnc(NCC2CC3CC3C2)[nH]1)C1CCN(C)CC1 C=C(C)CN=C(NCC1(Cn2ccnn2)CC1)N1CCC(COC(F)F)C1 C1(C(N2CCN(C(C34CCC(C3)OC4)=O)CC(O)C2)=O)CCc2ccccc2C1 CC1CNCCC1N.c1(C(=O)NC(C2CC(n3ccnn3)C2)=O)ccnc(CO)c1 N1(C(C=CC=C)=O)CCN(C(=O)C(C(C)C)NS(C)(=O)=O)CC1CC(=O)NC Cc1cc(F)cc(F)c1NC(C1CCN(C(c2ccc(F)cc2F)=O)CC1)=O N1(C(c2csc(C(=O)OC)c2)C(=O)NC)CC2CCCC12 C1(C)(C(=O)NC(c2cnn[nH]2)C)CC(=O)N(C)C1 c1(C(N2C(C)C(NC(c3cccs3)=O)CCC2)=O)nc2cc(O)ccc2[nH]1 N1(C(CCCSc2ccc(C)cc2)=O)CC(C2(NC(C3CCC(O)C3)=O)CC2)C1 C(=O)(CCCC(F)(F)F)N1CCC(C(=O)NCc2ncc(C(C)C)o2)CC1 c1(C(=O)NC2CS(=O)(=O)CC2NC(C2CCCCC2)=O)cccc2sncc12 c1(C(=O)OC)cc(Br)c(NC(=O)NC(C)C(=O)Nc2cccc(Cl)c2)c(I)c1 c12ccc(cc1)C(=O)NC2.c1(CC)cc(C(N2CCCC2CC)=O)no1 C1(NC(C2C(OC)CN(C(=O)OC(C)(C)C)C2)=O)C=CC(C)(C)CC1 C(=O)(C1=C(C#N)CCC1)NC(COCC)C(=O)N(CC(=O)NCC)C S(=O)(=O)(c1ccc(NC2CCC(=O)NC23CCC3)nc1)NC(CCCC)(C)C c1(CC)nc(NCC2C3CN(C(=O)CCCCN(C)C)CC23)c(C#N)cc1C C1(C2CCCO2)(C(=O)NCCCCCNC(c2cc3n(c2)CCC3)=O)CCCO1 CCCCC(CC)CN=c1nc(N(C)Cc2nocc2Br)cc(C)[nH]1 c1(CCC)cc(C(=O)NCC(C)(C)CN(C)C(C2(NC(N)=O)CC2)=O)cc(O)n1 C(CC(C(=O)NC1CC(O)CC1O)NC(c1ccc(O)nn1)=O)OC C1(CC)CCN(C(=O)CCC(C)NC(c2cc(C)c[nH]2)=O)CC1 c1(C(N2CCC(NC(C3N(C)CCOC3)=O)(CF)C2)=O)ccc(Cl)cc1Cl C1(N(C)C)(CC)CCN(C(=O)CCN(C(=O)C(C)n2cnnn2)CC2CC2)C1 c1(-c2nnc(C)o2)ccc(C(N2CCC2CNC(=O)C#CC2CC2)=O)cc1 c1(CC)nc(C)n(C)c1C(=O)NCC(CCOC)NC(c1cc(C(C)=O)cs1)=O Cn1ncc(C(=O)NC2CCCCC2NC(=O)Cc2ccnc(O)c2)c1N c1(C(=O)NCCC(C)NC(C=CCOC)=O)ccc(C(=O)NC(C)C)cc1 c1(OC)ncnc(C)c1C(=O)NCCCCCNC(c1c(C)cccc1Br)=O N1(C(c2c(OC)cc(C)cc2)=O)CCN(C(c2c[nH]nc2C)=O)C2CCC12 N1(C(CNC(=O)OC)=O)CCC2CCN(C(C3(Sc4ccccc4)CC3)=O)CC12 N1(C(c2c(OC)cccc2)=O)C2CC=C(C(=O)N3CCC(C)(CO)C3)C1CC2 c1(CC)cccc(C(=O)NC2(CNC(C3CCCN3C(C)=O)=O)CCOC2)c1O C(CC(=O)N1CCCC(CC2CNc3ccccc32)C1)(C(F)(F)F)OC Cc1cc(C(N2CC3CC3(C(=O)N(C34CCC(CC3)CC4)C)C2)=O)cc(C)c1 c1(OCC(=O)NC(C)CN(C)C(C2CC2Br)=O)cccc([N+](=O)[O-])c1 CCCC(C)(CC)C(=O)N1CCC(C(=O)NCC(c2ccccc2)C)O1 C1(NC(C2CCN(C(CC)=O)C2)=O)CC2(CCC(NC(=O)C(O)C(C)C)CC2)C1 C(C(=O)N1CC2(CCCO2)C1)(C(C)(C)C)NC(C(C)C#N)=O C1(C)(CC)COCCC1NC(=O)NCc1cc(C)cc(=O)o1 c1(C(=O)NC2C=CC(CNC(C3(N(C)C)CCC3)=O)C2)ccc2sc(=N)[nH]c2c1 c1(C(=O)OCC)cccc(Cl)c1Nc1c(C(N2C(SCC)CCCC2)=O)scc1 c1(C(=O)NCC2N(C(CC(c3ccc(F)cc3)C)=O)CCC2)ccc(C#N)cc1 C1(C(=O)NC2(C#C)CC2)CCCCC1(C)NC(=O)CC(C)(C)OC c1(CNC(C(CCNC(=O)Cn2cnnn2)O)=O)c(F)cncc1F c1(C(N2CCC(C)C(NC(c3cc(O)nn3C)=O)C2)=O)sc2nccnc2c1N N1(C(C=C(C)C(F)F)=O)C2CCC1C(CNC(C1CCC(C)(O)CC1)=O)C2 Cc1csc(C(=O)NC2(CNC(=O)C(C3CCCCC3)O)CCOC2)c1Cl C(CNC(=O)C(N1CCNC1=O)C)(C(=O)NCCC(F)F)OC c1(OCC(=O)O)ccc(CN2CCN(Cc3n[nH]cc3Br)CC2)cc1 C1(C(N2CCN(c3ccccc3)CC2)=O)CSCCN1Cc1ccc(Cl)cn1 C12(CC(N3CCC(NC(C4CC(C(C)C)OCC4)=O)C3)=O)CCC(CC1)OC2 C1(C)(CCNC(C=CC=CCC)=O)CCN(C(=O)C(O)CN2CCCC2)C1 C1(NC(c2c(OC)n(C)nc2)=O)CCN(C(C2(CCOC)CC2)=O)CC1O C(c1cccc(Cl)c1)=C(C)C(=O)NCC(C(C)(C)C)NC(=O)CC12CCCC1C2 Cc1nnc2cc(N3CC(F)(F)CC3(C)CNC(=O)C=Cc3cccs3)ncn12 n1(COC)nccc1S(=O)(=O)NC(C(=O)N(C)OC)C1CCOCC1 N1(C(C(CC)c2ccccc2)=O)CCC2CC(NC(=O)C(C)(C)O)CCC2C1 C(C(CC(C)C)NC(=O)CCCc1cnn[nH]1)NC(CCc1c(C)ncs1)=O c1(C(=O)NCC2C(NC(c3c(CC)occ3)=O)C2)coc2cc(F)cc(F)c12 C(=O)(CCCCC(F)F)N1C(CC)C(NC(c2cc(C(C)C)cc(F)c2)=O)CC1 C1(NC(C2C(COC)C2)=O)CC=CCC1C(=O)Nc1ccsc1C(C)C c1(CC(C(=O)NC(CN2CCC(OC)C2)=O)C)ccc(F)cc1 c1(COC)cccnc1C(=O)NC1CN(C(=O)C(N2CCSCC2)C)CC1C c1(COC)cc(C(=O)NC(CNC(=O)CCN(S(C)(=O)=O)C)C2CCC2)c(C)o1 N1(C(c2c(CC)c[nH]n2)=O)CC(NC(c2coc(Br)n2)=O)CC1(C)C C1(CC(=O)N(C(C)CN(C)C(C)=O)C)(OC)CCC1 CN1C(=O)CCC1C(N1CCC(C2CCCCN2C(c2ccsc2Cl)=O)C1)=O C1(CNC(COCCSC)=O)(CNC(C2CCC(=O)O2)=O)CCOCC1 c1(OC)ncc(C(=O)NC2CCC2CNC(c2cscc2C#N)=O)cc1Cl c1(OCC)ccc(CNC(=O)CCC2C(=O)Nc3ccccc32)c2ccccc12 c1(C(=O)NCC2CC(NC(CC3C(C)CCC3)=O)C2)ccc2c(c1)C(=O)C(=O)N2 c1(C(=O)OC)ccc(NC(C(=O)OC)C(C)O)c(Cl)c1 C(=O)(CCCC(C)NC(c1c(C)nn(C)c1N)=O)NCCCSC CCC(CC)C(=O)NC(C)CC1CN(C(=O)C(C)C(=O)OC(C)(C)C)C1 CCCC(C)CCCC(=O)N(CCCCCNC(c1sc(C(C)C)nc1C)=O)C N1(C(CC2CC(SC)C2)=O)CCOC2(CCN(C(c3c(CO)n[nH]c3C)=O)C2)C1 N1(C(CCOCCN(C(c2c(C)nc(O)cc2)=O)C)=O)CCOCC(C)(O)C1 C1(S(C)(=O)=O)(C(=O)NCC(CC)NC(c2cc(CO)c(C)o2)=O)CCCC1 N1(C(C(C)OC2CCCC2)=O)CCN(C(C2(n3cncn3)CC2)=O)CC1CCO CN1C2CCC1CC(C(N1CCC(NC(C3(C)CC=CCC3)=O)C(O)C1)=O)C2 c1(NC(C)=O)ccc(C(N2CCN(C(C3CC(O)CN3)=O)C3CC23)=O)c(C)c1 c1(CCC)nn(C)c(OC)c1N(Cc1ccc(OC)cc1)Cc1c(C)nn(C)c1C Cc1c(Br)cc(C(=O)NC2CC2CNC(=O)CC2CCOC2)cc1[N+](=O)[O-] C(=O)(C1CCc2cccc(=O)n21)NCCC1CCCN(C(C2(CC)CC2)=O)C1 N1(C(c2c(CC)n(C)nn2)=O)CCC(C)N(C(=O)C(C)CC(F)(F)F)CC1 c1(OC)ncc(C(=O)NCCc2ccc(C)s2)cc1C1=C(C)CCCC1 C1(C)(NC(C(N2CC(OCC)C(C(C)C)C2)=O)=O)CCC(=O)N(C)C1 CCCCCC(O)CC(=O)NC(C)CCCNC(=O)C=CC1CCCC1 C1(C)(CNC(NCC2(OC)CCC2)=NCCCOC)COc2ccccc2O1 N1(C(c2cn(CC)nn2)=O)CCC(C(=O)NCC2(CF)CC2)CC1 Cc1cc2sc(C(=O)NC3CC4CC(NC(=O)CCCF)C3C4)cc2s1 c1(C(=O)NCCCNC(C(C)=C2CCC2)=O)cccn(C2CCC2)c1=O Cc1ccc(F)c(N)c1C(=O)NC1CCOCC1NC(C1(C2CC2)CC=CC1)=O C(=O)(CS(C)(=O)=O)NCC1C(NC(CCCOC(CCC)=O)=O)COC1 N1(C(C(=O)N(C2(c3ccccc3)CCOC2)C)=O)CCN(CC(N)=O)C(C)(C)C1 c1(C(N2CCCC(NC(=O)Cc3nc[nH]n3)CC2)=O)cccc2nc[nH]c12 c1(C(C(=O)OC(C(=C)Cl)=O)C2CC2)ccc(C)cc1 C1(O)(CN2CCC(NC(Cc3cc(C)n(C)n3)=O)C2)CC(C)CC(C)C1 C1(CC(=O)N(CC(C)(C)NC(=O)C(F)(F)c2ccnn2C)C)CCCCC12CC2 C1(C(N(C2CCCCC2)CC)=O)CC2(C)CCC1(C)O2.c12cccc(c1)NC2=O CC1(NC(c2cc(-c3ccccc3)ns2)=O)CCN(C(=O)Cc2cncnc2)C1 CC1(C)CN(C(c2ncccc2O)=O)CC1NC(c1ccn(CC(F)F)n1)=O C(CCC(=O)NCC1CCN1C(C1(c2ccccc2)CC1(F)F)=O)NC(=O)C1CC1 N1(C(=O)C=Cc2ccc(Br)s2)CC2(CCCN(C(=O)C(F)=C3CCC3)C2)C1 CC1(C)CCCCC(C(=O)NC2CCCC(NC(c3cocn3)=O)C2)C1 CCCCCCC(C)CC(=O)NCC1CCN1CCNc1cn(CC)nn1 C1(CNC(C2C(CNC(c3csc(O)n3)=O)C2)=O)CC(O)C(O)C1 C1(CNC(=O)CNC(c2ccsc2)=O)CCCCN1C(=O)CN1CC2CC2C1 C#CC1CN(C(=O)C(C2CC=CCC2)NC(=O)CC=Cc2ccccc2)CCO1 c1(C(=O)NCC(=O)NCC2CC2NC(=O)C(C2CC2)C2CC2)cccc(F)c1 Cc1nc(C(=O)NC23CC(C2)N(C(=O)Cc2ccc(F)c(F)c2)C3)ccc1C#N c1(NC(N2C(CCCC)CCC2)=O)cnc(COC)nc1 Cc1c[nH]cc(-c2ccc(CN=c3[nH]c(C(C)(C)C)cs3)cc2)c1=O N1(C(=O)C=CC2CC2)CCC2CN(C(C3(F)CC3c3ccccc3)=O)CC12 c1(C(N2C(CNC(C3CC34CCSCC4)=O)CCCC2)=O)ccc2nn[nH]c2c1 S(=O)(=O)(c1cccc(C(=O)NC2CN(C(=O)C(C)C(=O)OC)CC2C)c1)NCC=C N1(C(=O)CCCOC2CCCC2)CCN(C(=O)Cn2cc(F)ccc2=O)C2CC12 c1(C(N(CC(C)NC(C(CCC)C#N)=O)C)=O)c(C)c2ccc(F)cc2oc1=O Cc1ccc2c(c1Br)CCC2NS(=O)(=O)CCOC1CC1C.C(C)(C)(C)O C1(NC(C(c2ccn(C)n2)(C)C)=O)COCCN(C(c2ccnn(C)c2=O)=O)C1 c1(C(=O)NC2(C)CN(C(=O)C(=Cc3cccnc3)F)C2)cnc2ccnn2c1 CC(CCNC(N1CCCCC1(C)CO)=O)S(=O)(=O)c1ccc(Cl)cc1 C1(C(=O)NCC2(F)CC(CNC(Cc3c(C)n(C)cn3)=O)C2)CC(C2CC2)=NO1 CCCCC(F)(F)C(=O)NC(C)C=CC(=O)NOCCCF Cc1ccnc(C(N2CCC(C3CCCCN3C(=O)CC(C)C)C2)=O)c1N Cc1n[nH]c(C)c1C(C)C(=O)NCC1C(C)CCN1C(c1cncc(Cl)c1)=O CC(C)(C(=O)Nc1nc(Cl)ncc1Cl)C(F)(F)F C(=O)(CCCS(N)(=O)=O)NC1C(NC(C(C(C)C)n2ccc(C)c2)=O)CC1 C1(OC)CN(C(c2c(C)ncn2O)=O)CC1NC(c1cc(Br)n(C)n1)=O N1(C(c2c(CC)c[nH]n2)=O)CCN(C)CC1C(N1CCC(n2cccn2)C1)=O N1(C(C2(CC=C)CCC2)=O)CC2(CC(C(=O)Nc3ncccc3CC)CO2)C1 C1(NC(c2cc(C)sc2)=O)CCCC(C(=O)NCCCC2CC(C)C2)CC1 N1(C(CC(CCC)O)=O)CCC2(CCC(CNC(=O)C(F)=CC3CC3)OC2)CC1 C#Cc1ccc(C(=O)NC(CN(C)C(c2oc(Br)cc2C)=O)CC)c(C)c1 C1(NC(c2cc(C)ncc2)=O)CC2CC(NC(C3(F)CCCCCC3)=O)C2C1 C=CCC(C)(C)CC(=O)N1CC2CCCC1C2C(=O)Nn1cccn1 c1(C(C)NC(=O)Nc2ccc(C(=O)OC(C)(C)C)nc2)nsc2ccccc12 c1(-c2cn(C3CC(C(C(C)CCCCO)=O)C3)nn2)cc(F)c(F)cc1F C1(N(C)C(=O)OC(C)(C)C)(C(=O)NC(c2ncnn2C)C2CC2)CC(CO)C1 c1(NC2CCN(c3nnc(C(N)=O)o3)C2)cc2ccsc2[nH]1.C12CCN(CC1)C2=O C1(NC(C2CC=C(C)CC2)=O)CCN(C(=O)Cc2ccc(O)cc2Cl)C1(C)C C1(O)(CNC(CN2C(C)CC2)=O)CN(C(c2csc(CS(C)(=O)=O)n2)=O)C1 CCC(CC)(CO)C(=O)N1CC2CCC(C(N3CCCCC(SC)C3)=O)(C2)C1 C1(C(N(CCO)CC)=O)CCN(C(=O)CC2COCC(C)O2)O1 N1(C(CN(CCC)C)=O)CCOC2(CCCN(C(=O)C(C)CO)C2)C1 N1(C(c2noc(C)c2C)=O)CCC12CN(Cc1ccc(C(F)(F)F)nc1Cl)C2 CC(C)(C(=O)OC(C)(C)C)C1=CCN(C(=O)C(F)CC(Cl)Cl)CC1 C1(CC(=O)OC)CC(C(=O)OC)CN(Cc2ccc(C(=O)OC)o2)C1 C1(CNC(c2nc(CC)sc2)=O)CCCN(C(=O)C(c2cnccc2C)(C)C)C1 O=C1NC2(CO1)CC(C(N1CC3CN(C(c4cn(CCO)nn4)=O)CC3C1)=O)C2 C1(COC)(NC(c2ocnc2C)=O)CCN(C(=O)C(C)OCC(C)C)CC1 CCC(CC(C)C)C(=O)N1CC(O)(CN(C(=O)CCC#N)Cc2ccccc2)C1 C1(C)(NC(CCOCCCOC)=O)CCN(C(C2(O)CC2(C)C)=O)CC1 CC1CN(C(c2c[nH]c(=O)cn2)=O)CCC1C(N1CCC(N=[N+]=[N-])C1)=O c1(C(=O)NC23CC(NC(c4cnc(-c5ccccc5)[nH]4)=O)(C2)C3)ccc(=O)oc1 N1(C(C(CC(C)C)C)=O)CCn2ncc(CNC(=O)CSCCC(F)(F)F)c2C1 O(NC(=O)C(CNC(=O)C(C)N(C)C)OC)CC#C CN1CCC(C(=O)NC(CNC(c2coc(Oc3ccccc3)n2)=O)CO)C1=O c1(C(N2CC(NC(c3ccc(F)cc3Br)=O)C(F)(F)C2)=O)ccc(F)c(Br)c1F c1(N(CCN(C)C(c2ccc(C(F)F)cc2F)=O)C)[nH]c(=O)n(C)c(=O)c1C#N Cn1c(=O)cc(C(N2CCN(C(=O)C3=CCCC3)C(CO)C2)=O)c2ccccc12 Cc1cc(C(N2CC(CNC(=O)CC3CCCC3C)C2)=O)[nH]c1C#N C#Cc1ccc(C(=O)NC(CNC(c2n[nH]cc2F)=O)C2CC2)cc1Cl Cc1cnc(C(=O)N(CCCC(=O)NCC(C)C(C)O)C)c(F)c1 c1(C(=O)NC(C(=O)NCC(CSC)OC)(C)CO)cc(C)nnc1C c1(C(N2C(CN(C(C3C(C(C)C)(CC)C3)=O)C)CCC2)=O)cncc(C2CC2)c1 C#Cc1c[nH]nc1C(=O)NC1C2CC(NC(C3CC3CC(C)C)=O)CC12 Cc1cc(C(N2CC(F)(CNC(=O)C(C)C=Cc3ccccc3)C2)=O)nn1C CC(=O)C(C)CC(C)C(=O)N(C)CC1CCCCN1C(C1CNC(=O)O1)=O C(=O)(CCCCCC#N)N(CCCNC(C(CC1CCCCC1)OC)=O)C c1(-c2cn(CCC3CN(C(c4oc(CC)c(C)c4)=O)C3)nn2)ccc(Cl)c(F)c1 C12(C(=O)NCCCCCNC(=O)Cc3ccccc3F)CSCC1C2(F)F C1(C(=O)OC)CCC(C2CCCCC2)CN1c1nccc(=NCC2CC(O)C2)[nH]1 C1(C(=O)NCC2CC(NC(C3(CO)CCCO3)=O)C(O)C2)(CC)CC(F)(F)C1 C1(C(=O)NCCNC(=O)C2CC2)(CC)CN(C(c2ccncc2)=O)C1 N1(C(CCN(CC)CC)=O)CCC2(CCCN2C(=O)CCC2=CCCCC2)CC1 N1(C(N2C(CCC)COCC2)=O)CC(C)N(C(C)C)C(C)C1.c12nn(C)cc1N2 C1(NC(C2CN(C(C)=O)C2)=O)CC2CCC(C1)N2C(=O)CCCCN(C)C C(C)(C(C)COC)(c1nnnn1CCSC)NC(c1scc(CC)n1)C N1(C(c2c(OC)csc2)=O)CCCC(CNC(c2ccc(C(C)=O)cn2)=O)C1 N1(C(C2(CC=C)CC2)=O)CCC2CCCC(C1)N2c1ncnc2sc(CC)cc12 N1(C(=O)C(F)CC2CCOC2)CC(N(C(=O)CC2(O)CCC2)CCO)C(O)C1 C1(C(=O)NCC(n2cc(CC(CO)C3CC3)nn2)C)CN2CCN1CC2 N#Cc1cc(C(=O)NC(Cc2cc(Cl)sc2Cl)CO)cc(Cl)c1 N1(C(C(CCC)NC(C2C=CCS2)=O)=O)CCC2(CCCN2C)C1 O=C(CCCCNC(=O)C(C1CCCCC1)O)NC1(C(F)(F)F)CCC1 c1(C(C)(C)C(=O)NC2CCCC2C#N)ccc(F)cc1Br C(=O)(C(O)CC(F)F)NCC(C1CC1)NC(c1ccc(CC(C)C)cc1)=O CC1CC(C(N2CC(OCCF)C2)=O)N(C(C23CSCC2C3)=O)C1 C1(CNC(C2N(C(C=C(CCC)CCC)=O)CC(O)C2)=O)CCC(C)(C)CO1 CC1CCC(C(=O)NC2CC3C(C2)C3(F)F)CN1C(c1cncn1C)=O c1(C(N2CC(CNC(C(c3cnn(C)c3)OC)=O)C2)=O)sc2ccsc2c1C CC1=C(C(=O)N2CCN(C(c3c[nH]c(C(N)=O)c3)=O)C3CC23)SCCO1 N1(C(c2c(C)oc(CO)c2)=O)CC(NC(C2C(F)(F)C23CC3)=O)CC1(C)C c1(C(=O)Nc2c(C)cc(NC(c3nccn3C)=O)cc2)cc(F)c(Cl)nc1Cl C1(N(C(C=CSC)=O)C)CN(C(c2cc(C)cc(C)c2)=O)CC12CC2 Cc1nc(=NC(=O)C2(F)CCN(C(c3ccc(-n4cnnc4)cc3)=O)C2)s[nH]1 C1(CNC(c2scc(COC)c2)=O)CCN(C(C2CSCC(=O)N2)=O)C12CC2 N1(C(CC2(C=C)CC2)=O)CCC2(CCN(C(c3cncc(OCC)c3)=O)CC2)C1 CC(CC1CCOCC1)C(C(=O)NCCN1CCOCC1)N1CCCCC1CF C1(CNC(=O)CC(F)F)CN(C(c2cc[nH]c2)=O)C2CC12 c1(C(N2CCC(N(CC(O)C3CC3)CCO)C2)=O)cccc(F)c1F Cc1nnc(CCNC(=O)COC(C)(C)CNC(=O)Cc2cnnn2C)s1 C1(CNC(Cc2cc(C)ns2)=O)CC(NC(c2cccc(CO)c2)=O)C1(C)C C1(NC(CCC#C)(C)c2nnnn2C2CCC2)CCc2ccccc2NC1=O CCC(C(=O)OC)C(=O)N1CCCN(C(=O)NC2C3CCC2CC3)CC1 c1(C(N(C2CCN(C(C3CC3F)=O)C2)CC)=O)nc2ccccc2[nH]1 C1(NC(c2cncc(CC)c2)=O)CC(O)CN(C(=O)C(c2cccc(C)c2)F)C1 C1(C2CN(C(C(C)SC)=O)C2)CN(C(=O)CCCCF)CCO1 C(=O)(CC(C(=O)NC1(CNC(=O)C(=O)NC2CC2)CCC1)NC(C)=O)OC CC1CCC(c2cn(C3CC(C(=O)NC(F)C(C)C(F)F)C3)nn2)CC1 c1(C(=O)Nc2c(C)nc(Cl)nc2)cc(-c2ccc(C(C)O)cc2)cc2[nH]ncc12 Cc1c(C(=O)NC2CCCC2CNC(c2cnn(C(C)C)c2)=O)cccc1F C1(C(=O)NCC2CC3CN(C(CCOC(C)C)=O)CC32)CN2CCCN1CC2 C(=O)(C(C)(C)CN(C)C)NCC(CC)NC(=O)CCCCc1cnn[nH]1 c1(C(N2CCN(C(C(C)=C(C)C)=O)C(CCO)C2)=O)ccc(Cl)c(S(N)(=O)=O)c1 c1(C(=O)NCC(CNC(=O)Cc2ccc(O)nc2)OC)cncc(C2CC2)c1 C1(CC=C)(NC(=O)CCc2ccc(C)nc2)CCN(C(=O)Cc2ccn(C)c2)C1 C(=O)(C(Cn1ccnn1)NC(=O)C(OC)OC)NCC1CC(CC)C1 C1(CC)(NC(=O)CN(C)C(C)C)CCCN(C(c2ccnn2C(F)F)=O)C1 C1(N(C)C)CCC(CNC(C2(C)CN(C(=O)C(F)F)C2)=O)CC1 Cc1cccc(OC(C)C(=O)NCCOCCNC(c2c(C)[nH][nH]c2=N)=O)c1 C1(C)(CNC(c2cc(C)nnc2)=O)CN(C(=O)COCC(F)(F)F)CCO1 CC(C(C)(C)C(=O)NCC1(C)C=CCCC1)NC(=O)CC1CC1 C1(C(=O)NC2(CC=C)CCN(C(=O)C(C)SC(C)C)C2)(OC)CCCC(C)(C)C1 CC(C)C(C(=O)N(C(C)C(N)=O)C)C(C)NC(C1CN(C2COC2)C1)=O Cc1ccc(C(=O)N(C)C(c2cccnc2)C)c(C(F)F)c1 C1(C(=O)NCC2(C(N)=O)CN(C(CCCNC(N)=O)=O)C2)CCN2CCOCC12 c1(OC)nccc(C(=O)NC(C)CCN(C(=O)CN2CCCCCC2)C)n1 c1(C(=O)NCCC(C)NC(C2N(CC)C(=O)CC2)=O)ncn2ccccc12 Cc1cccc(C=CC(N2CCCC(CO)(NC(C3CCC(C)(C)C3)=O)C2)=O)c1 c1(C(=O)NC(C2(O)CN(C(=O)C(C)S(N)(=O)=O)C2)C)cc2c(cn1)OCCC2 C(=O)(CC(C)Cc1ccc(Cl)cc1)NCC(C)N(C(COCCC)=O)C c1(SCC)cnccc1C(N1CCC(CO)(CNC(=O)C(C)CC)C1)=O n1(CC(N2CCC(N)(Cc3ccccc3)C2)=O)ccc2nc(O)nc(O)c12 N1(C(C(C)C#N)=O)CCC(NC(c2c(Cl)cccc2Br)=O)C(C)(C)C1 C=CC(CCC)CC(=O)NCC1CN(C(c2nn(C(F)F)cc2Cl)=O)CCN1C c1(C(=O)NCC(C)(C)OCCNC(=O)CSS(C)(=O)=O)cc[nH]c(=N)n1 CC1CC(C(=O)NC2CC(C(C)NC(=O)C=C3CN4CCC3CC4)C2)=NO1 c1(SCC(=O)NC2(C)CC(NC(C(C)OCCC=C)=O)C2)ccc(C(C)C)cc1 C1(NC(COCCCCC)=O)CS(=O)(=O)C2CN(C(=O)C(C)(C)CF)CC12 c1(-c2ccnc(OC)c2CO)ccc2c(c1NCc1ccc(Cl)o1)OCO2 c1(C(N2C(C(C)NC(Cn3ncc(CC)c3)=O)CCC2)=O)nccnc1C C1(NC(C(c2cccc(C)c2)C)=O)CC2CCC(C1C)N2c1ncc(Cl)c(O)n1 C(CC1=CCN(C(=O)C(F)(F)c2cnn(C)c2)CC1)NC(Cn1ccc(C)n1)=O Cc1cccc2c(C(=O)NCCCNC(C3CC(CF)C3)=O)c[nH]c12 c1(C(C(=O)NC2N(C(COCCC)=O)CCOC2)OC)cc(F)cc(F)c1 N1(C(CCC(C)O)=O)CCC(C2CCCN(C(C3(CO)CCC3)=O)C2)CC1 N(C(=NCc1sccc1OC)NC1CCOc2ccccc21)CCOCC c1(C(N(C2CN(C(c3c(C)coc3)=O)CC2(C)C)C)=O)cc(F)c(F)cc1F c1(C(=O)NCC2(C(C)(C)O)CN(C(C3(C(C)(F)F)CC3)=O)C2)csc2nccn12 Cc1nc(O)nc(C)c1CC(=O)N(C)CCN(C)C(c1cc(Br)cnc1N)=O N1(C(CC2(CC)CCC2)=O)CCC(CNC(C2C=C(C)CS2)=O)C1(C)C c1(OC)cccc2c1OCC(C(=O)NCC(F)CNC(=O)CS(=O)(=O)N(C)C)C2 CCC(CCC(=O)N1CCN(C(=O)C(=Cc2cccc(Cl)c2)C)CC1CF)OC C1(CNC(c2cc(CSCC)on2)=O)CCN(c2cc(F)ncn2)CC1C c1(C(=O)NC(C)CN(C(=O)CC2CCCCC2(C)C)C)cc2cncn2c(O)n1 c1(C(=O)NC2(C)CN(c3nc(C)nc(Cl)c3)C2)cnn2ccn(C)c12 N1(C(C(C)(C)OCCC)=O)CCC(C(=O)NCC(c2cnn(C)c2)O)(CC)C1 c12cnc(cc1OC)Nc1cc(C(=O)OC)ncc1-2.c1(OCC)cc(SC)on1 N1(C(CCC(C)(F)F)=O)CCCN(C(c2cncc(O)c2)=O)CCC1 C(=O)(C#CC1CCOCC1)N1CCCC(NC(CC(C)C(C)(C)C)=O)C1C CC#CC1CCN(C(c2ccccc2C)C(=O)NCCC2CC2)C1 C12(C(=O)NCCCSCC)CC1CN(C(=O)C(C1CCC1)OC)C2 N1(C(C2CC(OC)CN2C(=O)CC2CC2)=O)CCN(CCO)C(=O)C1 c1(C(=O)NCC2(NC(C3C(OCC)CC3)=O)CCCCC2)cc(O)cc(Cl)c1 c1(OC)cc(Br)cc(NC(C2C3CC2N(C(c2cccc(CO)c2)=O)C3)=O)n1 C#CC1(C(=O)NC2CC(Cl)C2)CCN(C(=O)CC2CCOC2=O)C1 c1(Nc2c(C(=O)OC)cc(OC(F)(F)F)cc2)ccccc1S(=O)(=O)C(F)F CC1(CS(=O)(=O)Nc2ccc(N3CCC(N)CC3)nc2)CCCCC1(F)F C1(CN(C(c2nc(CC)sc2)=O)C)CN(C(=O)C(O)CC)CC12CC2 N1(C(=O)CN2C(=O)CNC2=O)CCCC(C2CCN(CCCC(F)(F)F)CC2)C1 c1(C(N(CC(C)NC(=O)Cc2ccc(F)cc2F)C)=O)ccc(F)c(CO)c1 N1(C(CN2C(C)CC2)=O)CC23CC1(C2)C3.C1(C(N)=O)CCOCC1 Cc1ccsc1C=CC(=O)NCCC1CC(NC(C2CCCCO2)=O)C1 Cc1nnc2n1CC(C(=O)NC1(CO)CN(C(=O)C(C)OCC(F)(F)F)C1)CC2 CCC(CC(=O)NC1CCCCC1O)NC(C1CS(=O)C1)=O C1(NC(c2c(C)c(C3CC3)on2)=O)CC2CC1CN(C(=O)C(C)C(F)(F)F)C2 CC(C)CC(CC(=O)NC(C)CCO)NC(C1CCCCC1)=O C1(C)(COC)CC(NC(c2ncoc2C(C)C)=O)CN1C(=O)CSC(C)(C)C C1(CNC(C2CCN(C)C2)=O)CCC12CCN(C(c1cc[nH]c1C1CC1)=O)CC2 C(=O)(CC(CC)CC(C)C)NCC(CCC)NC(=O)COc1ccsn1 c1(NC(C(C2CCN(C(c3ccc(C#N)cc3)=O)CC2)C)=O)c(Cl)cccc1Br c1(C(=O)NCCCNC(C2C(C)(COC)C2)=O)ccccc1ON(C)C C(=O)(C(O)CC(F)(F)F)NS(=O)(=O)CC1CN(C(CC(COC)COC)=O)C1 n1(CC(=O)N(C(C)CCC#N)CCO)nnn(-c2cccs2)c1=O C(=O)(CCN=C(NCC1CCOC1)N(C)Cc1cc(C)nn1C)NC c1(CC(=O)OC)ccc(CC(=O)NCCNC(=O)C=C2CCCC2)cc1 c1(C(=O)NC2CCN(c3nc(SC)nc(C)c3)C2)ccc2c(c1)C(C)CN2 C1(C(=O)NC(c2ccc(Cl)cc2)CO)CCCC(NC(c2ccnc(Cl)n2)=O)C1 N1(C(CCSCC(N)=O)=O)CCCCCC(NC(c2cnc(Cl)[nH]2)=O)C1 CN1C(=O)NCC12CN(C(C1CCCN(C(c3ccc(F)cc3)=O)C1)=O)C2 C(=O)(C(Cc1ccco1)C(=O)N(C)CCN(C(=O)C(C)c1cncs1)C)OC C1(C(=O)NCCCOCCC(=O)NC(C(C)C)(C)C)C2CCCOC12 N1(C(=O)Cn2cc(CO)nn2)CCC2(CCCN2C(C2(CCF)CC2)=O)C1 c1(OCC)ccc(C(=O)N(CC)CC2CC2)cc1Cl.C1(C(C(=O)N)C)CCOCC1 C1(C(N(C)Cc2nc(C)on2)=O)CC12CCN(C(c1scnc1C)=O)C2 C1(NC(c2snc(Cl)c2Cl)=O)CCCN(C(=O)C2=CCCC2)C1 C(=O)(C(C)(C)CC(F)F)NCC1C(NC(CCNC(=O)NC)=O)C1 N1(CCC)CCC(C(=O)NC2C3CCN(C(c4cccc(CSC)c4)=O)C23)CC1 N1(CC(CO)NC(c2ccsc2Br)=O)CCCCC1 C1(O)(CNC(C(C)NC(C)(C)C)=O)CCN(C(c2ccc[n+]([O-])c2)=O)C1 Cc1c(C(=O)NCC(C)NC(=O)CCOC(C)CC(C)C)ccn1C CCCC(O)C(CO)NC(C1(CNC(c2ncnc(O)c2F)=O)CCCC1)=O CC(CC(=O)N(CCCNC(c1cn(CCCF)nn1)=O)C)NC(N)=O C1(C(N2C(C3(O)CN(C(c4cc(Cl)ns4)=O)C3)CCC2)=O)CCc2nnnn2C1 C(CN=c1[nH]c(=NCC2Cc3ccccc32)c2[nH]ccc2[nH]1)OC(=N)O C=CC1(C(=O)NCC(C)(O)C2CCC2)CCN(C(=O)C(O)C(F)(F)F)CC1 C1(NC(C2CCN(C(=O)NC)CC2)=O)CCCN(C(c2c[nH]c(CO)c2)=O)C1C c1(C(=O)NCCCNC(CCc2cncc(C)c2)=O)cc(C)nc2ccccc12 c1(OCC)ccc(SCC(=O)NCCC(C)NC(=O)Cc2ccnn2C)cc1 C=CC1CN(C(=O)COC2CCCCC2)CC1NC(=O)CC1CCN(C)C1 CCCC(F)(F)C(=O)N1CC=CC(NC(=O)Cc2ccnn2C)C1 c1(N2CCCC(OC)C2)nc(=NCCc2conc2Br)[nH]c2c1CCC2 c1(NC(C2(F)CCN(C(Cc3nc(C)on3)=O)C2)=O)cc(F)ncc1F C1(NC(CCC(=C)C)=O)CC(OC)CN(C(C2CC(=O)N(c3cn[nH]c3)C2)=O)C1 CS(=O)(=O)c1cccc(NC(c2cc(Cl)cnc2-c2ccc(F)c([N+](=O)[O-])c2)=O)n1 C=CCC(CC(=O)NC(c1cscn1)C)NC(C1CCC1(F)F)=O C(=O)(C(CNC(=O)Cc1ccc(F)nc1)CC1CC1)NC1C(C(=O)OC)CC1 N1(C(c2c(C)c[nH]c2)=O)CCCC2(C1)CN(C(c1ccc(NC=O)cc1)=O)C2 C1(NC(C2(C)CC(=C)C2)=O)CCN(C(=O)COC2CCOC2)CC1F Cc1cc(C(=O)NCC(CO)NC(c2cnc(N(C)C)o2)=O)c(C)n1CC1CC1 S(=O)(=O)(c1ccc(CCC#N)cc1)NC(CCN1C(C)CCC1)=O c1(CNCC(c2ccc(S(C)(=O)=O)cc2)(C)O)cc2c(Br)cccc2o1 C(=O)(CS(=O)(=O)N(C)C)NCCN(C(=O)Cc1cccc(C(N)=O)c1)CCOC c1(N(CC(CNC(C(CC)CC(F)F)=O)C)C)ncc(Cl)cc1[N+](=O)[O-] C=CC(O)(C(=O)N1CCC(C(=O)N(C2(CO)CCCC2)CCCC)CC1)C(F)(F)F C1(C(N(C)CC2(OC)CCCC2)=O)CCN(C(=O)CC2CCCC(=O)C2)CC1 C1(C)(C(=O)NC2CC(N(C(C(c3cnccn3)C)=O)C)C2)CC2(CCC2)C1 Cc1c(C(=O)NCCCNC(=O)CC(O)CN(C)C)cccc1[N+](=O)[O-] CCC(CC)C(=O)NCCCCCNC(=O)C(c1cccc(F)c1)C C1(C(=O)NC(C2CCCN(C(C3CC(N=[N+]=[N-])C3)=O)C2)C)CS(=O)(=O)CC(=O)N1 Cc1cc(C(=O)NCCNC(C2SCCS2)=O)nn1C(F)F C1(C(=O)N(CC(F)(F)F)CCO)CCCCCN1C(=O)C(Cl)Cl C1(CC(=O)NC(CC)CNC(C2(C(N3CCCC3)=O)CC2)=O)CCS(=O)(=O)CC1 C1(F)(CNC(=O)Cc2cccnc2)CC2CCC(C1)N2C(C1CC(=C2CC2)C1)=O Cc1nocc1CC(=O)NCCCCCN(C(c1sccc1Cl)=O)C(C)C CCN=c1[nH]c(C(=O)NCC2CC3CN(C(C4(C)CCCCO4)=O)CC23)cs1 N1(C(C(CCC)F)=O)CCCCCC1C(=O)Nc1cccc(OC)c1O Cc1cc(F)c(Cl)cc1C(=O)N(C)CCN(C)C(c1cnnn1C1CC1)=O c1(C(=O)NCC(CC)NC(C2COC3(CO)CC2C3)=O)nn(C)c(C)c1Br C1(C(=O)NCCCCN(C(C(C(=C)C)(C)C)=O)C)CC12CCC(C)(C)CC2 N1(C(CSCC#C)=O)CC2CCCCC2(CNC(C2CC(=C)C2)=O)C1 c1(C(=O)NCCN(C(C=CC(C)C)=O)CCN(C)C)cnn(C(F)F)c1 c1(OC)cc(C(=O)NC2(CC(=O)NCC3CC34CC4(F)F)CCCCC2)ccn1 C1(C(=O)Nc2ncc(C)c(I)c2)COC2(CCN(C(=O)CCC(F)(F)F)CC2)C1 C1(C2N(Cc3nnc(C(C)C)s3)CCC2)CCCN(C(c2cc(Cl)ncn2)=O)C1 c1(C(c2n(CC)nnn2)NCc2cncc(C)c2)n[nH]c2ccccc12 C1(C(=O)NC2(C)CC2)CC12CCN(C(C1CC13CCCCC3)=O)CC2 C1(N(C(=O)CCN2CCC2)C)CCCCN(C(c2ccc(Br)c(N)c2)=O)C1 C(C(F)(C(=O)NC(C)Cc1nncn1C)C(C)C)NC(CC(C=C)(C)C)=O N1(C(C2(C#C)CN(C(C3CC(N(C)C)C3)=O)C2)=O)CCCC(N(C)C)CC1 N1(C(C2(CC)CCCC2)=O)CCOCC(NC(C2CCC2(OC)OC)=O)C1 c1(CC(C(=O)O)NC(=O)NC2CC(C)(CO)C2)csc2ccccc12 C1(CC(=O)NCC(N(C(CCC=C)=O)C)C2CC2)CCC2(CCC2)O1 C1(NCC(C2CCOC2)C)COCCC1C(=O)NCC(F)(F)F N1(C(CCC(C)=O)=O)CCC(O)C(C(=O)NC(c2ccc(F)cc2)C)C1 C(=O)(C(C)(C)CN(C)C(C1COCCC1C)=O)NCC(C)CO CCC(CC(C)C)C(=O)N1CCC(NC(c2cnc(OC)s2)=O)C1(C)C c1(-c2cn(C(c3ccc(C)o3)NCC3CCCS3)nn2)nn2c(c1C(=O)O)CCC2 C(=O)(CCCC(F)(F)F)NCC1CCCN(C(C(CC)C(=O)OC)=O)CC1 c1(N(C(c2ccc3nsnc3c2)C(=O)NC2COC2)CC)ccc2c(c1)OCO2 C1(C(N2C(C)CCC(NC(c3cnc(S)nc3)=O)C2)=O)CC2(CCCC2)CO1 N1(C(C)(C)C)CC2CC(C1)C2O.c12ccnc(c1)N(C(=O)CC1CCC1)C(=O)CC2 C1(CC=C)(C(=O)NC(C)C(=O)OCC)CCCN1C(=O)Cc1cccnc1O c1(C(C)NC(=O)NC2(CCOC)CCOC2)ncccc1F Cc1nc(C)n(CC(N2CCC2CNC(C2(CS(N)(=O)=O)COC2)=O)=O)n1 c1(C(N(CC(C)N(C(CN(CCC)C)=O)C)C)=O)cc([N+](=O)[O-])nn1C N1(C(=O)C=Cc2ccncn2)CCCC2(CCN(C(=O)Cc3c[nH]nc3O)C2)C1 c1(N2C(C)CC(NC(=O)COCC3CCOC3)C2)nc(O)c2ccccc2n1 Cc1noc(C)c1CCC(=O)N1CC(NC(=O)Cc2nnn(C(C)(C)C)n2)C1 C=CCC(C)C(=O)N1CCCCC1CCN(C(=O)CC(C)(F)F)C C1(C(N2CC(CCNC(C=CCOC)=O)C2)=O)CCCCC1C1CC1 C12(C(N3C(C(=O)Nc4n(C)nnc4)CC4CC43)=O)CC3CC(CC(C3)C1)C2 N1(C(C(C)CN(C)C)=O)CC(CNC(c2cnn(C)c2N)=O)OC(C)(C)C1 N1(C(C2N(C(C3(CC)CC3)=O)C(C)C2)=O)CCCCC(CO)C1 C(=O)(C1=CCCC1)NC1(C(=O)NC2CCC(SC)C2)CCCC1 c1(N(C(c2ncsc2C)C(=O)NC)CCCOCC=C)ccccc1OC C1(NC(C2CN(C(C3(O)CCOCC3)=O)CCO2)=O)CC2(CCCCC2)C1 C1(CNC(c2ccc(C(C)(C)C)[nH]2)=O)CCCN(C(C2(CF)CC2(F)F)=O)CC1 CCC(C)(C)CC(=O)N(C(C)C(=O)Nc1cccc(OCF)c1)CC C(N=c1[nH]nco1)C1(NC(C(c2cncc(F)c2)C)=O)CCCC1 Cc1ccnc(NC(=O)NCCC(C)OC(=O)NC(C)(C)C)n1 Cc1nc(Cl)cc(=NC(C)C2CN(C(C3(O)CCSC3)=O)CCO2)[nH]1 Cn1nc(C(=O)NC2CN(C(C3(O)CCC3)=O)CC2C(F)F)c2c1CCCC2 c1(OC)cnnc(OC)c1C(=O)NC1CC2CN(C(=O)CSS(C)(=O)=O)CC12 Cc1cc(C(=O)NC2(C)CC(C(=O)NCCOC3CCCC3)C2)cs1 c1(C(=O)NC2CCN(C(c3ccc(C)c(Cl)c3)=O)C(C)C2)ccc(F)c(F)c1F C(=O)(C(C)(C)CCCNC(c1cncs1)=O)NC(C(N(OC)C)=O)C C(C(O)CC(C)(C)O)N1CC(OC)(CO)C1 C(c1cnc[nH]1)=CC(N1CC(O)(C2CCCN2C(C2CCCOC2)=O)C1)=O N1(C(=O)Cc2cccnc2F)CCC2(CC1)CC(N1CCCCC(O)(CF)C1)C2 CCCCC(C(=O)NCc1ccsc1C(=O)NCCC(F)=C(F)F)N(C)C C1(C(=O)NCC(C)NC(C2CCOCC2(C)C)=O)CC12CCc1ccccc12 C1CC2=CCN(C2)C(=O)C(C)O1.C=CCN(CC=C)CCSC Cc1c(NC2CCN(CCCO)CC2)ncnc1NC1CC(C(N)=O)C1 N1(C(C(CCSC)NC(=O)Cc2ccco2)=O)CCC2(CCC(O)C2)C1 N1(C(C(CC2CCCCC2)OC)=O)CCC(CNC(c2ccc(C)s2)=O)CC1 C1(CNC(C2CCN(C(CC)=O)C2)=O)COC(C)(C)CN1C(C1(C)COC1)=O N1(C(CCCCC=C)=O)CCC2OCCN(C(c3ccc(=O)n(CC)c3)=O)C2C1 CNS(=O)(=O)N1CCC(C(=O)NCC2COC3(C)CC2C3)CC1 N1(C(C(CC)(C)CNC(=O)C(C)CC(F)(F)F)=O)CCC2CC1C(=O)N2C C=CC(CC)CC(=O)N1CCC(OCC2CCN(C(=O)Cn3nccn3)CC2)C1 c1(C(=O)NCC2(O)CCCN(C(C=COCC)=O)C2)ccc2c(C#N)c[nH]c2c1 C(=O)(C1=NOC(C)(C)C1)NCC1C(C)CN(C(=O)C=Cc2ccnn2C)C1 C1(C)(CN(C(COC(C)C)=O)C)CCCC1NC(C1CNC(=O)C1)=O c1(-n2ncc(C(N3CC(NC(C4(CF)CC(=O)C4)=O)C3)=O)c2)ccccc1C#N CCCCCCCCCC(c1nnnn1CCCOC)NC1C=CCCCC1 c1(OCCC(=O)NCC(CC)NC(=O)CC2COCC2O)ccc(C)c(C)c1 c1(C(=O)COC(c2cc(-c3ccncc3)on2)=O)c(OC(F)(F)F)cccc1F C(CC(=O)NC(C)CCNC(c1c(Cl)n[nH]c1C)=O)(C1=CCCC1)OCC n1(CC)ncc(C(=O)NCC2(F)CN(C(c3nccnc3C)=O)C2)c1Cl c1(C(=O)NCC(CCCC)NC(=O)CSCCC)cncc2c[nH]nc12 Cc1ccc(C)n1CC(N1CCC(NC(c2ccc(F)s2)=O)C1C)=O Cc1nn(CCC(=O)N(C2CCCC(NC(C3(O)CC3)=O)C2)C)cc1Br C(C(C)(C(C)C)NC(c1nnn(CC)c1C)=O)NC(CCOCC)=O C1(C(N(C)CCc2cnccn2)=O)(CNC(=O)Cc2ccns2)CC12CCC2 C1(CCC(=O)NCCN(C(=O)C(c2ccccc2)N(C)C)CCC)CCCCO1 c1(C(=O)NCC23C(CN(C(CN4CC(C)C4)=O)C2)C3)cc(Cl)cc(Br)c1 C1(NC(CCCNC(C)=O)=O)CCN(C(c2cnns2)=O)CC1(C)C N1(C(c2c(CC)ocn2)=O)CC2(CCN(C(=O)C(CC)SC)CC2)C1CC Cc1ccc(SCC(=O)NCCC2CCCN2C(=O)C(C2CCOCC2)C)cc1 c1(-n2c(CCCN(C)C)nc(-c3ccnc(Cl)c3)n2)ccnc2c1cnn2C C#CCC(C)(C(=O)NCc1ncc[nH]1)NC(=O)Cn1ncn(C)c1=O C1(F)(C(=O)NCCOCCC(=O)NC(c2nccn2C)CC)CCC(C)CC1 N1(C(c2c(OCC)cccc2)=O)CC2(C)CN(C(C3CCNC3=O)=O)CC2(C)C1 N1(C(C(C)CC(N)=O)=O)CCC2(CC(NC(C3CCNCC3)=O)CO2)C1 c1(C(N2CCCC(CNC(=O)Cc3ccsc3)C2)C)ccc(Cl)cc1 C1(NCCC2(C#N)CCC2)CCN(CCc2ccc(F)cc2)CC1 c1(C(N2CC3(C(NC(COCC#C)=O)CC3)C2)=O)ccc2nc(O)[nH]c2c1 FC1(F)CCc2onc(CN=C(NCC(F)=C(Cl)Cl)NCC3CCCO3)c2C1 c1(C(N(C2CCN(C(c3cnn(CC)c3)=O)C2)CC)=O)cc(Cl)cnc1C C(=O)(CC(C)C(C)C(C)C)NCC1OCCCN(C(Cc2cccc(C)c2)=O)C1 C(=O)(CC(C)(C)CC(=O)OC)NC1CCCCN(C(C2(CC=C)CCC2)=O)C1 C(C(O)CC(=O)N1CCC1(C)CC(=O)NCCC1(O)CCC1)N(C)C CC(Cc1ccccc1)C(=O)N(C)CCOCCNC(C1CC1F)=O C1(NC(c2nc(CC(C)C)sc2)=O)CCC2CN(CCC3CC=CC3)CC2C1 C1(C(N(OC)Cc2ccc(Cl)cc2)=O)CCCC(CN)N(C)C1 C1(O)(CNC(C(C=C)O)=O)CCCN(C(c2n[nH]c(C3CC3)c2Cl)=O)C1 S(=O)(=O)(c1cccc(F)c1)N1CCCC(C(N2CCC23CCCOC3)=O)CC1 C1(C(=O)NC2CCCCC2CNC(=O)C2=CSCCO2)(OC)CCCCCC1 C(CCCCC(=O)N1CCC(OCCNC(C2CCC(F)C2)=O)CC1)=CC c1(C(N2CC(CCNC(C3C(C(C)(C)C)C3)=O)C2)=O)cncc(CO)c1 C(=O)(C(C)CCCc1cn(C(C)C(=O)O)nn1)Nc1ncc(C)cn1 CCCCCC(F)C(=O)NCCCCC(C)NC(c1cnc(C(C)C)nc1)=O C1(OC)(CNC(=O)C(F)=C(C)C)CN(C(C2(Cl)CC2(F)F)=O)C1 C1(C2CCN(C)CC2)(C(=O)NCC2(C)N(C(C(C)OCC=C)=O)CCC2)CC1 C1(CC)CN(C(=O)CC(N)C(C)(C)O)CC2(CCOC2)O1 N1(C(C(C=C)(C)CC)=O)C2CCC1CC(CNC(C1CC1C1CC1C)=O)C2 N1(C(CNC(CCSC)=O)C(F)F)CCN(C(=O)COC2(C)CCOCC2)CC1 N1(C(C(F)=CC)=O)CCN(C(=O)CCc2cccc(CC)c2)C(C)C1C N1(C(C2=CC(C)(CC)C2)=O)CC2(CCN(C(=O)C(C)(C)CC3CC3)CC2)C1 N1(Cc2c(C)noc2C)CCC(C)(C(=O)Nc2cnncc2Br)CC1 c1(C(N2CC3C(CNC(c4ccc(C)cc4Cl)=O)(C3)C2)=O)ccc2ncnn2n1 N1(C(CNCCCC)=O)CCOCC(C(=O)NS(=O)(=O)C(F)F)C1 c1(C(=O)NC(CCNC(C(c2ccccc2)NC(COC)=O)=O)C)cccnc1 N1(C(CC2OCCN(C(C(c3cn(C)nc3)=O)=O)C2)=O)CCC(O)CC(C)(C)C1 c1(C(=O)NCC2CC(NC(C(C)N(C(C)=O)C)=O)C2)cc(Cl)ccc1F C1(CNC(CC(C=C)(C)C)=O)CCC2(CCC2)C1NC(c1cccc(Cl)c1)=O Cc1cc(C(N2CC3(C2)CN(C(=O)C(O)CC2CCOCC2)C3)=O)cc(O)c1 Cc1nc2cnn(C)c2cc1C(=O)NC1CCCN(C(C2CC2(F)F)=O)CCC1 CCN=c1[nH]c(C)c(C(N2CCC(CNC(=O)CC3CCCO3)C(F)(F)C2)=O)s1 C1(N(C(=O)CCc2cn[nH]c2)C)C2CN(C(c3nc(C(F)(F)F)cs3)=O)CC12 Cc1ccncc1CC(=O)NC1(CNC(=O)CCCC2CCCCC2)CCC1 C1(CNC(c2ccc(C)cc2Cl)=O)C(C2CC2)CCN1C(c1snc(O)c1Cl)=O c1(CN2CCC(CC(=O)NCCCC3CCCCC3)C2)cc(Cl)c(Cl)cc1Cl c1(C(=O)NC2CCN(C(C3CC3(F)Cl)=O)C2)cc(=O)cc[nH]1 C1(C)(NC(C(N2CCCC(C)C2)=O)=O)CCC(NC(C2CCC2)=O)CC1 c1(CC)ccc(C(=O)NC2CCCC2NC(=O)C(O)C2CCC2)c(OC)c1 N1(C(c2ccccc2-c2onc3c2CCCC3)=O)CCC2(CCCNC2)CC1 CC1CCN(C(c2cnc3n2CCS3)=O)C(CNC(C2(O)CCCC2)=O)C1 C1(C(=O)NC(CC)C(=O)OC)CC(O)CCN1C(=O)C=Cc1cnc[nH]1 C(=O)(C(F)(F)c1cncs1)NCC(C)(C1CC1)NC(CSCCN(C)C)=O c1(OC)cc(C)c(Cl)cc1C(N1CCC(NC(=O)C(C)(C)n2cccn2)CC1)=O O=C(C1=CCSC1)NC1CC(CNC(C2(Nc3cccc(O)c3)CC2)=O)C1 c1(COC)cc(F)c(S(=O)(=O)N2CCCC(C(F)(F)F)C2C)c(F)c1 c1(C(=O)Nc2ccc(C(=O)OCC)o2)ccccc1CCN1CCC(C)CC1 c1(C(=O)NC2(C)CN(C(C3CCOC(C)(C)C3)=O)C2)cc(N=S(C)(C)=O)ccn1 C1(C(=O)NC(CCN(C(Cc2cc(C(=O)OC)sc2)=O)CC)C)CC=CCC1C c1(C(=O)NCCC(C)NC(c2ccnc(OCC)c2F)=O)ccc2cnoc2c1 C1(C(=O)OC)CC(NC(c2cccc(-c3ccccc3)c2O)=O)CC(C)(C)O1 C1(CC(=O)NC)CN(C(c2ccnc(SC3CC3)c2)=O)CCN1C(=O)CC(C)F Cc1cc([N+](=O)[O-])cnc1C(N1CCN(C(C2CCOCC2)=O)CC1CF)=O C(CC(C)C)(C(=O)NC(c1nc[nH]n1)CO)ONC(COC)=O C1(CNC(C2CC23CCC3)=O)CC2(CC2)CN1C(c1cc(C(F)(F)F)on1)=O C1(C(=O)NCC2(F)CC(NC(C(CC=C)NC(C)=O)=O)C2)CCCC(F)(F)C1 c1(C(N2CCN(c3ccc(C(=O)OC)cc3)CC2)=O)ccc2c(c1)CCCO2 c1(C(N(CCCCO)C(C)C)=O)ccc(CNC(C2COC(C)C2)=O)o1 CCCCCCCNCc1ccccc1N1CCN(C)CC1 C1(CC)C(C(=O)NCC(Cl)C(C)(F)F)CCN1C(=O)CSC(C)C c1(CC(=O)NCC2C3CN(C(C4(C(F)(F)F)CCC4)=O)CC23)ccc(Cl)cc1 c1(NC)cnc(C(=O)N(CCCNC(C2(C3CCCCO3)CC2)=O)C2CC2)cn1 c1(N2CCC(C(C)O)C2)nc(N2Cc3ccc(Cl)cc3C2)nc2c1CSC2 CC1(C)CC(O)(C(=O)NCC2CCCC(CNC(c3cnc(C#N)s3)=O)C2)C1 C1(C(=O)NCC(c2ccccc2)N(C)C(c2ccccn2)=O)OCCN(C)C1=O C(CC(=O)NC1CC1)(CC(N1CC(OCCc2ccn(CC)c2)C1)=O)OCC CN1C2CCC1CN(C(C1CN(C(C3(CO)CCOC3)=O)CC13CC3)=O)C2 C1(=CC(=O)NCC(CCNC(C(CC)C(F)(F)F)=O)O)CCOc2ccccc21 O=C1CCc2ccc(C(=O)NCc3ccc(C4CCCNC4)cc3)nc2N1 c1(C2C(C(CN(C3(C#C)CCC3)C)=O)C2)noc2c1CCCCC2 C(=O)(CCCCCCN=[N+]=[N-])NCCC(C)NC(c1ccc2nc(S)oc2c1)=O CC(C)C(F)C(=O)NC(C(=O)NC1(C)CC2(CC2)C1)C1(C)CC1 C(CCOC)(C(=O)NCCCCC(C)C)NC(c1cc(OC)no1)=O c1(C(=O)NC2C(CNC(CNC(N)=O)=O)CCCC2)ccnc2ncccc12 C1(C)(NC(C(Cn2cncn2)NC(C(C)N(C(C)=O)C)=O)=O)CCC(C)(C)C1 C(C(CN=c1[nH]c(Cl)nc2c1SCC2)C(F)(F)F)NC(Cn1c(C)c(Cl)cn1)=O CC#CCC(C(=O)NC(CCO)C(F)F)NC(c1cc(C)nc(O)c1)=O C1(NC(c2ccc(C)nc2)=O)CCC(C)N(C(=O)C=Cc2cn(C)nn2)C1 Cc1c(N)ccc(C(N2CC(NC(c3ncc(F)cn3)=O)C3(CCC3)C2)=O)c1Cl C1(C(=O)OCC)CCCN(Cc2ccc(O)cc2)C12CCC2 Cc1cc(Cl)c(Cl)cc1C(N1CCC(O)(CN(C(=O)COCC2CC2)C)CC1)=O C1CCC(=O)N(CC2CCC2)CC1.C1(C(=O)NC)CC(OC(=O)C(F)(F)F)CN1C(C)=O N1(c2n(CC)c(CCc3noc4ccccc34)nn2)CCC(C2(O)CC2)CC1 CCCCCCC(C)C(=O)N1CCN(C2CN(C(C3(C)CCCN3C)=O)C2)CC1 c1(NC(C23C(CN(C(C4CCN(C)C4)=O)C2)CC3)=O)cnc2cccnn12 C(=O)(C(C)(C)C(O)C(C)C)NCC(C(C)C)NC(c1cc(O)cc(O)n1)=O C(=O)(C1CCCc2nc(C)[nH]c21)NCC(C)(C(C)C)NC(C)=O C1(CC(=O)NCC2(O)CC(NC(=O)C(O)CC3CCCCC3)C2)CCCCCC1 CC1(CNC(=O)CNC=O)CN(C(c2sccc2Br)=O)CCO1 c1(C(=O)OC)cc(C(=O)NCC(O)CN(C)C(c2ccc(CF)cc2)=O)c(C)o1 CC(CCN=c1nc(CC2CC2)[nH]s1)NC(c1sccc1-n1ccnn1)=O C1(O)(CC(=O)NCCc2cc(C(N(CC(C)C)C)=O)no2)CCCOC1 C1(C(=O)NCC2CCN2C(=O)C(CO)N2CCCCC2)CN2CCC1CC2 C1(CC)CN(C(=O)CCn2cnc(C)cc2=O)CCC1NC(c1cc(Cl)no1)=O c1(C)cn(CC(=O)N(C2CCCCC2)CC(=O)OC)nn1.C1(C=O)C(C)CC1C N1(C(C(N2CCOCC2)C)=O)CCCCCC1C(=O)NCC(F)C1CCC1 C1(NC(CCCC=C)=O)COC2(CCN(C(c3ccc(CC4CC4)cc3)=O)C2)C1 c1(C(=O)NC2CN(C(c3c(C)cnnc3)=O)CC2C)sccc1S(=O)(=O)N(C)C N1(C(Cc2cc(C)sc2)=O)CCC(CF)(NC(C2CCOC(C(C)C)C2)=O)C1 Cc1cc(C(=O)NC2(CN(C(=O)CC3CCN(C)C3=O)C)CC2)c(C)n1C(C)C Cc1nc(CCC(N2CCOC(CNC(=O)C(c3ccncc3)C)C2)=O)oc1C C1(C(N2CCCC(C(N3CCN(CCO)CC3)=O)C2)=O)(CC)CCCCO1 C=CC1(C(=O)NCCC(C)N2CCC2)CCN(C(=O)CCCC(=C)C)C1 CC1(C)CCC2(CC1)CN(C(=O)C(F)C(F)(F)F)C2 CC1(C)NC(=O)N(CC(N2CC(NC(=O)CC3CCCCCC3)C(F)C2)=O)C1=O c1(C(N(C(CNC(CC(CCC)(C)C)=O)C)C)=O)cnn2ccc(Cl)c(F)c12 C1(NC(=O)Cc2csc(Cl)c2)CCN(C(C23CCCC2C3)=O)CCC1(F)F C1(NC(C2C(=C)C2)=O)CN(C(c2ccccc2-n2cccc2)=O)CC1(C)C c1(C(N2CCC(C)(NC(CC3(C=C)CCC3)=O)C2)=O)ccc2cc(C)ccc2c1 CCCCCC(C)CC(=O)N1CCCCC1CNC(C1CC2(CCCO2)C1)=O C(=O)(C1Cc2ccc(F)cc21)NCC1N(C(c2cnc(C)[nH]2)=O)CC1 C1(NC(=O)COC2CCN(C(C3CCCCCC3)=O)C2)CCCCCC1CO c1(OC)cc(C(N2CC(NC(c3cc(=O)c(OC)c[nH]3)=O)C2)=O)cc(Cl)c1 c1(C(CC)(O)CN(C(C)CN2CCCCC2)C(=O)NCCO)ccc(F)cc1 C1(NC(=O)COC2CCCCC2)CCN(C(c2cnn(C3CCC3)c2)=O)C12CC2 c1(C(=O)NC(C2CCCN(C(=O)OC)C2)C)ccc2c(c1)CCOC2 S(=O)(=O)(c1ccc(NC(c2ncc(C)o2)C)c(C#N)c1)NCC(CC)OC C(C1=CCCN(C(c2cnn(C(C)(C)C)c2)=O)C1)NC(c1c(OC)scc1)=O C1(NC(CCc2cc(C)[nH]n2)=O)C=CCC(C(=O)NCC(F)(F)CC2CC2)C1 N1(C(CCC2N(C)CCCC2)=O)CCC2(CC1)C(NC(=O)CCF)CS2(=O)=O c1(SC)nc2ncnc(NC3(C4CCN(C(=O)CC5CC=CC5)CC4)CC3)c2s1 C(CC(=O)NCCOC1CN(C(=O)CCNC(N)=O)C1)N(CCC)C Cc1[nH]nc(C(N2CCOC(C(=O)NCc3ccco3)C2)=O)c1O N1(C(C23CCC(OC)C2C3)=O)CCN(C(c2cc(O)nc(O)n2)=O)C(C2CC2)C1 N1(C(CCC)=O)CCC(C2CN(C(=O)Cc3csc(SCCN(C)C)n3)C2)CC1 C1(C)(CNC(C(Cn2ccc(C)n2)C)=O)CN(C(c2c(O)noc2C)=O)CCO1 C=Cc1cc(C(N2CCC3(NC(=O)CCCNS(C)(=O)=O)CC3C2)=O)cc(F)c1 C(N=c1nc(N2CCN(CC=C(C)C)CC2)cc(C)[nH]1)c1ccc(CCC)c(F)c1 C(=O)(C1CCCc2sccc21)NCC1CN(C(C2C3(CC(C)(C)C3)C2)=O)C1 c1(C(=O)NCC2(O)CN(C(=O)C=Cc3cncs3)C2)ccc(F)c(Cl)c1F N1(C(c2nc(C(C)C)sc2)=O)CCC(NC(C2(CF)CC(F)(F)C2)=O)CC(O)C1 c1(CNC2CCC(C(=O)NCc3cn(C(C)C)nc3)C2)c(Cl)cccc1Cl C1(C(=O)NC(CC=C)C)CCC(F)(F)CC1 C=CCC(CC(=O)NCC1CC2COCC2C1)NC(=O)C=CC(C)CC N1(C(C2(CC)CCC2)=O)CC2CC(C)N(C(c3cc(C)c(C)cc3C)=O)C2C1 C1(NC(c2ccc(CC(=O)OC)n2C)=O)CCC12CCC1(CC2)OCCO1 CC1CC(NC(=O)CC2COCC(C)O2)CN(C(=O)CC(=O)OC(C)(C)C)C1 c1(C(=O)NCc2nnc(C3CCCOC3)o2)cc(F)c(Cl)cc1F CC(C)(C)CC(F)C(=O)N1CC(c2ccncc2)C1.C12CC(C1)N2 S(=O)(=O)(c1cc([N+](=O)[O-])cc(Cl)c1F)Nc1c(-n2ncc(C)c2)ccnc1 S(=O)(=O)(c1cc([N+](=O)[O-])ccc1C)N1CC(CNC(c2c(C)ncc(C)n2)=O)C1 Cc1cc(C(=O)NCC2CCN(C(C3CCC(F)(F)C3)=O)C2)nn1C1CC1 c1(CNC(=NCC)NCC(c2ccc(F)cc2)O)nc(Br)c(C)cc1Cl C1(NC(C2CC=C(C)CC2)=O)C2CC1N(C(C1CCC(N(C)C)CC1)=O)C2C c1(N2CC(C)(c3ccccc3)OCC2)ccc(Br)c(S(=O)(=O)N2CCCC2CO)n1 C(=O)(C(C)(C)C(=O)N1CCC(C(C)(C)CNC(C2CC2(F)Cl)=O)CC1)OC c1(N2CC(NS(CCOCC)(=O)=O)(CO)C2)ncnc2[nH]cc(C)c12 C=CC(CCC)CC(=O)NC(CC(C)(C)C)C(=O)NC1CCC(C)(C)C1 C(F)(F)(C(F)C(F)(F)F)Oc1ccc(NCCc2cc(COC)ns2)cc1 N1(C(c2cc(C)n(C)c2)=O)CCC(C)N(c2cc(C(C)C)nc(Cl)n2)CC1 C#CC1(NC(C2(NC(C3CCCC3C(C)C)=O)CC(CO)C2)=O)CCC(C)(C)C1 c1(C(=O)NC2C(CNC(C(CC)OC3CCCC3)=O)C2)cc(OCC)ccc1Cl N1(C2CCN(C(COCCC#C)=O)C2)CCC(NC(c2sncc2)=O)CC1 N1(C(C2=CC(C)(C)C2)=O)CCC2(C=C(C(=O)N3CCCOC(CO)C3)C2)C1 CCCC(C(=O)N1CC(CCNC(c2conc2COC)=O)(OC)C1)OC C1(C(=O)NC(CC=CC)CO)CCN(C(=O)COCCCOC)CC1(C)C CC1(C)COC(C(=O)NCCC2CCN(C(=O)Cn3cc(Cl)cn3)C2)CO1 C(CCCCC(=O)N(CCNC(c1cc(O)cc(F)c1)=O)CC)=CC CC(C)(O)CCN=C(NCc1sccc1Br)NC1CCCC1 c1(NC(C2(NC(C3CCO3)=O)C(C)C2)=O)cc(CO)cc(F)c1 c1(NC(c2cncc(NC(c3c(C)ccs3)=O)c2)=O)ccc2c(c1)C(=O)CCC2 C1(OCC(=O)NCC(C2CC2)NC(c2n(CC#C)ccc2)=O)CCC(F)(F)CC1 Cc1cc(C(=O)NCC2CCCN2C(=O)C(C)(C)N2CCCC2)cc(Br)c1C N1(C(CCC=C)=O)CCCC(C2CCCNC2)C1 C1(N(C(CNC(C2C(C)C2)=O)=O)C)CC2CCC(C1)N2C(=O)CCn1cccc1 c1(C(CN(C2CN(C(=O)NC3CCCC(OC)C3)C2)C)=O)ccc2c(c1)CCC2 C(c1ccc(F)c(Cl)c1)=CC(N1CCC(C)(NC(c2cc(C)cc(Cl)c2)=O)C1)=O c1(C(=O)NC2CC(O)(CNC(CSCC)=O)C2)cnccc1C CC1CN(C(=O)CCCC2CC2)CCN1C(C1(O)CCCCC1)=O c1(NC(C(CC2CC2)NC(c2ccsc2)=O)=O)ccc2n[nH]cc2c1 Cc1cc(CCC(=O)NCC(=O)NCC(=O)NC2CCC2C(N)=O)on1 C1(NC(CC2C=NN(C)C2=O)=O)CN(C(=O)CN(C2CCSC2)C)CC1C1CC1 CCCC(CC)CCC(=O)NCC(C)CNC(=O)CCc1nccn1C C1(=CC(=O)NC2C(NC(C(CC)Sc3ccccc3)=O)C2)CCC(C)CC1 C1(C(=O)NC2C(NC(CC3CCC(C)(C)CC3)=O)C2)CC2CSCC(C1)C2 Cc1[nH]c(C)c(C(N2CCCC(CCNC(=O)COc3ccsn3)CC2)=O)c1C N1(C(c2c(CC)csc2)=O)CCC2(CCCCN(C(=O)C(CC(C)(C)C)OC)C2)C1 C1(C(N2CCC3(C(NC(=O)COC4CCOC4)C3)C2)=O)CCCN2CCCC12 C12(NC(=O)COCC3CCCO3)CC3CC(CC1C3)C2.C12CCC1C(=O)N2 c1(C(N2CCCCCC2c2cccc(C)c2)C(=O)NCC=C)nc(Br)ccc1F C(=O)(CCC(CF)CF)N1CCC(C(C)C(=O)NCCOCCN(C)C)CC1 Cc1cc(Cl)c(C(N2C3CCC2C(NC(C2CC24CC4)=O)C3)=O)cc1C C1(NC(=O)CC2(c3ccccc3)CC2)COCCC1NC(c1csnc1C1CC1)=O CCCC(C#N)C(=O)N1CC(CC(F)C(=O)NCC(O)CC(F)(F)F)C1 CC1CN(C(=O)COc2ccc(F)nc2)CCN1C(C1(C)CCC(=O)C1)=O C1(CNC(COC(C)C)=O)CN(C(=O)CC2(CO)CC2)CCC1C Cc1c(F)ccc(C(N2CC(C)(C)CC2CNC(=O)CCCOC(C)C)=O)c1N C1(CNC(c2ccc(CC)o2)=O)CCN(C(=O)C=Cc2ccccc2C)C12CC2 CCCCC(O)CNC(=O)C(C)CN(C)C(c1nocc1CC)=O C(=O)(C(F)CC(C)(C)NC(c1c(OC)nsc1)=O)NC1CCC(C)(CC)CC1 c1(C(=O)NCC(CC(C)(C)C)O)coc2c1C(=O)NCCC2 c1(CC(=O)NC2CC3(C(C(N4CC5C(CC)(C5)C4)=O)C3)C2)cncc(C#N)c1 c1(CC)ccc(CC(=O)NC(CNC(c2nn(C)cc2C)=O)C2CC2)cc1 c1(SC)cc(C(N2CCCC2CCNC(C2CC3C(C2)C3(F)F)=O)=O)ccc1F C(=O)(CC(C)(C)C(F)F)N(C(CC(=O)N(C)Cc1ccc(CC)o1)(C)C)C c1(OC)cc(O)ccc1CNC1CC(C(C)C)N(C(=O)OC(C)(C)C)C1 c1(C(=O)NC2CN(C(CP(C)(C)=O)=O)CC(F)C2)ccnc2cc[nH]c12 c1(C(N(C(C(=O)NC(CC=C)C)C)C2CC2)=O)ncnc(O)c1F C(c1cccc2ccccc12)=CC(=O)NCC(C)(O)C(F)(F)F C1(CNC(N(C(c2ccc(Cl)cc2)C)C)=O)CCc2nn(C)cc2C1 C1(C(N2CC(N(C(CSCCOC)=O)C)C(O)C2)=O)Oc2ccccc2C1C N1(C(C(C2CC2)OCC)=O)CCN(C(c2cc(C(=O)OC)[nH]n2)=O)CC1 c1(C(=O)NC2CCC(NC(C3CC(C)(C)C3)=O)C2)csc(N=S(C)(C)=O)n1 c1(OC)nc(C(=O)NCC2CCC(F)(CN)CC2)ncc1F c1(N2C(c3ccccc3F)(CC)CC2)cc(Cl)ncc1C(=O)OC(C)(C)C c1(C(=O)NC2CCC(C)N(C(=O)C=C3CCCC3)C2)c(F)cc(C#N)cc1F N1(CC2CCC(C)O2)CC(NC(C2CCCN2c2ccccc2)=O)C(C)(C)C1 c1(C(N2CCCCC(N(C(C(CSC)C)=O)C)C2)=O)occ2c1CCOC2 C(CC(=O)NC1CC(CCNC(c2csnn2)=O)C1)SCC(C)C CON=CC(=O)NC1CC(F)(CNC(c2coc(-c3ccccn3)n2)=O)C1 C1(C(N(CC(CCC)C)C)=O)CCN(C(c2nn(C)cc2Cl)=O)C(C)C1 N1(C(Cc2ccc(C)s2)=O)CC2CC(NC(=O)CCc3cc(C)sc3C)C1C2 N1(C(CCOC(=O)NCC)=O)CCC(C2N(C(c3oncc3C)=O)CC2C)CC1 c1(NC(CC2(N(C)C(C3CCC(C4CC4)O3)=O)CC2)=O)cccc(Cl)c1 C1(N(C(=O)C(N2CCNC2=O)C)C(CC)=O)CC(NCCN2CCC2)C1(C)C C(=O)(C(COC)C(F)(F)F)NC1(CC)CCN(C(c2cnn(C)c2N)=O)CC1 c1(C(N2C(C)CC(NC(c3cn(C)nc3O)=O)CC2)=O)nc2ccccn2c1F N1(c2nc(C(=O)OC)c(C)s2)C(CNC(C2CC2C2CC2C)=O)CC2COCC12 c1(CC(N2C(CC)C(C)CC2)=O)cnn2c1CCCC2 C1(C)(NC(CC2N(C(c3ccc(OC)s3)=O)CCCC2)=O)CN2CCC1CC2 C1(NC(N(C)CC2CCC(F)(F)C2)=O)CCCCCC1n1cccn1 C1(CC(=O)NC2CC(NC(c3ccc(C)o3)=O)CC2O)CCCCC1(C)C N1(C(C(c2n(C)ccc2)=O)=O)CCCC(C2(NC(c3cnc(S)nc3)=O)CC2)C1 c1(OC)ccc(C=CC(=O)NCC(C)(O)CNC(C2CCC2C#N)=O)cc1 N1(C(C2(SC)CN(C(=O)C=Cc3cn(C)nn3)C2)=O)CCC(C(N)=O)CC1 c1(C(=O)NC(CC)CNC(=O)C(C)(C)OC)ccc(OC)c(OC2CCCC2)c1 n1(C(CC)C)cc(C(=O)N(C)CC2(CNC(C3CC(OC)C3)=O)CC2)cn1 c1(OC)cccc(C(N2CC(NC(C3(OC)CCC3)=O)C(C(F)(F)F)C2)=O)c1 C12(C(=O)NCC(CC)NC(C3(C)CCCS3(=O)=O)=O)CCC(CO)(CC1)C2 C1(CNC(=O)COCC2CC2)CN(C(=O)CCNc2ncccn2)C2(CCC2)C1 c1(CN(CC)CC)ccc(C(=O)NC(C)CCNC(=O)Cc2ccno2)o1 c1(C(=O)NCC#CCNC(CCn2ccc(C)n2)=O)sc(=N)[nH]c1C CCCC(CNC(c1ccc(Br)cc1)C1CC1)CCC CC1CN(C(=O)COc2ccc(C(N)=O)cc2)CCC1NC(C1CC(F)(F)C1)=O N1(C(C2N(C(C)=O)CCC2)=O)CC2(CCN(C(=O)CC3CC4CCC3C4)CC2)C1 C#CCCCC(C)C(=O)NCC1(O)CC(CNC(c2cccc3c2OCC3)=O)C1 c1(OC)ccc(OC)c(C(=O)CCC(=O)OCCCCC2(C)OCCO2)c1 C1(=O)CCCC2CC2NC(=O)CC2CCN12.CCC(CC1CCC1)c1cn[nH]c1 C#CCC(CC(=O)NCc1nn(C)c(=O)o1)NC(c1cccs1)=O c1(C(c2cnn[nH]2)NCC(=O)NC2CC(C(=O)OC(C)(C)C)C2)ccccc1 C1(O)(CN(C(=O)Cc2c[nH]ccc2=O)C)CCCN(C(C2CCCC(=O)N2)=O)C1 c1(C(N2CCC(C(C)NC(=O)CC(F)(F)F)C2)=O)cc2ccsc2s1 c1(OC)cc(C)ccc1CN(c1ncc(-c2cnn(CCC#N)c2)cn1)CC1CC1 C(=O)(C1CCc2nnc(C)n21)NCC(C)(C)NC(c1cc(C)[nH]c1C)=O C12(CNC(C=CCNC(CC#N)=O)=O)CCCN1CCC2 N1(C(C=COCC)=O)CC2CCC(C1)C2CNC(c1sc([N+](=O)[O-])cc1Cl)=O c1(C(N2CCC(O)(C(C)NC(CCC)=O)C2)=O)cc([N+](=O)[O-])cnc1N CCCCCCCCC(C)C(=O)NCC1CN(C(=O)COC(C)=O)CCN1C C1(C(N2CCOCC2)C(=O)NC(=O)NCc2n(C)nnc2)Cc2ccccc2O1 C=CCC(C)(CC)C(=O)NCC1C(CNC(c2c(C)coc2C)=O)C1(F)F C(=O)(C(F)(F)F)NCC(=O)NCCC1CN(C(=O)C(O)C2CC2)C1 C12CCN(CC1)C(=O)C(C)COC(=O)CC(=O)N2C1CC1.C(C)(C)(C)OC C(C)(CO)(CC(C)C)SCC(C(=O)OCC1CC(=C)C1)OC(C)(C)C C12(C(N(CC(CC)NC(=O)C3=COCCO3)C)=O)CCC(CC1OC)C2 C1(CC)C(C(=O)NC(COCC2CC2)CC)CCCN1C(=O)C#CC1CC1 c1(C(N(C)CC2CN(C(c3c(CC)nc(C)[nH]3)=O)C2)=O)noc2ccc(F)cc12 C(=O)(CCCCC(=O)N1CC2CCC2(CNC(=O)CCC2CCOC2)C1)OC C1(NC(C2C(C3C(C)C3)C2)=O)CC2CN(C(=O)CCCn3cncn3)CC2C1 n1(CCC(=O)N(CC(C)(C)C)CC(C)C)cc(C2CCCO2)nn1 C1(C(N2CC3C(CNC(C4CN(C5CC5)CCO4)=O)(C3)C2)=O)CC2C=CC1CC2 c1(CN2CC(O)(CNC(c3ccc(Br)c(Cl)c3)=O)C2)cc(Br)ccc1Cl C(=O)(C(O)CCCNC(=O)C(O)CN1CCCC1)N(C)CC1(C#N)CCCC1 CCC(C)(C)CC(=O)NC(C(=O)NCC1(C)CCN(C)C1)C1CCCO1 c1(CCC(=O)NC2C(NC(C(C)=CC)=O)CCC2)c(C)nc(S)nc1C c1(NC(CNC(c2ccc(OCC#C)cc2)=O)=O)cc(=NC2CC2)cc[nH]1 N1(C(C(C(CC)CC)OC)=O)CC2CCCC(C1)N2C(=O)C(C)S(C)(=O)=O CC(C)(CNC(=O)CN1CCOC1=O)CC(=O)N1CCC(O)C(CO)C1 c1(N(CCNC(=O)C#CC2CCCC2)CC)ncc(C#N)cc1F C1(C(=O)NCC(C2CCCC2)NC(CC2(C=C)CC2)=O)CCCC(=O)N1C c1(OC)ccnc(C(=O)NCC2CCCN(C(c3ccc(C(F)F)s3)=O)C2)c1O N(C1C(=O)N(C)CCc2ccccc21)C(=O)NCC(CC)Oc1cc(Cl)cc(Cl)c1 Cc1cc(-c2ocnc2C(=O)NCC2(F)CN(C(=O)CN(C)C(N)=O)C2)on1 N#Cc1cccc(CCC(=O)NCC(F)CNC(c2cccnc2C2CC2)=O)c1 CC1CCN(C(C2C3CCCC23)=O)C1C(=O)NCC1(F)CN(C)C1 c1(OC(CC)C)ccc(CNC(C)Cn2cc(CO)nn2)cc1 C(=O)(C(CC1CCC1)OC)NC1CC(C(=O)OCC)C1.C12CN(C1)C2=O C(CN=c1nc(C)cc(C)[nH]1)N1CCN(C(c2cncc(OC)n2)=O)CC1 c1(C(=O)NC2CCCN(C(C=C(CC)C)=O)C2)ccc(-c2ccncc2)c(F)c1 CC1CN(C(=O)C2=C(Cl)CCC2)CCN(C(C2(C)C(C)(C)C2(C)C)=O)C1 N1(C(Cc2cc(OC)no2)=O)CCC(C)C(NC(=O)CCN2CCC(F)C2)C1 N1(C(C2COCC(C)O2)=O)CCC(N=[N+]=[N-])(C(N2CC3(C2)CC(C)(O)C3)=O)C1 CCCC(C(=O)N1CCC(C(F)F)CC1)NC(=O)CC1(OC)CCC1 Cc1cnc(NC2(CO)CCCCC2)c(S(=O)(=O)NC2CC3CC(O)C2C3)c1 C(=O)(CC(C(=C)C)OCC)NCC(CC=C)NC(=O)Cn1cc(Cl)cn1 CS(=O)c1ccccc1C(=O)NCCC(O)CNC(=O)CCc1ccccc1 CC1(NC(c2cc(C(F)(F)C(F)(F)F)ccc2O)=O)CCN(S(N)(=O)=O)CC1 C12(NC(c3c(C)sc(O)n3)=O)CCCC(NC(C3CCCC3C)=O)(C1)C2 C(=O)(C1Cc2ccc(Cl)cc21)N1C2C(CNC(c3ccccc3)=O)C(C2)C1 C(N=c1[nH]c(C(c2ccccc2)(C)C)cs1)c1n(CC)nnc1Br N1(C(c2c(C)cc(C(F)F)o2)=O)CCC2(CC1)CC2C(=O)NCC(C)O C(COC(C)C)(C(=O)NC(C)(CNC(c1cc(C)[nH]n1)=O)C1CCC1)NC(C)=O CC1(C)CCN(C(=O)CC(C2CC2)NC(C2(C#N)CC2)=O)CCO1 C(=O)(CC(C(F)F)NC(C1(C(=O)NC)CCC1)=O)NC(CC(=O)OC)C1CC1 Cc1cc(F)cc(C)c1C(=O)NCC1(F)CC(NC(c2nocc2Cl)=O)C1 C#Cc1cccc(C(=O)NCC(C)CNC(c2nnn(C)n2)=O)c1 Cc1oc(C#N)cc1C(N1CCC(O)(CNC(=O)CC2CC2C)CC1)=O c1(OC)cc(C=CC(N2CC3CCOC3(CO)C2)=O)ccc1OCC(N)=O CC(CCO)C(=O)NCCCCCn1cc(CS(=O)(=O)CC)nn1 n1(CCC(=O)N(C(CNC(C(C)CF)=O)C)C)c(=O)oc2cc([N+](=O)[O-])ccc12 c1(C(N2CCC(CCO)C2)C(=O)NC(C)C)cc2c(Cl)nccc2s1 N1(CCc2ccn(CC(C)C)n2)CCCCC1c1nc(C(C)C)no1 CN=c1[nH]cc(-c2cccc3nc(C(=O)Nc4cc(C)nn4C)cn23)cc1C#N Cc1cc(C)c(C(N2CCC(CO)(NC(c3cccc(C)n3)=O)CC2)=O)cn1 c1(C(=O)NCC2CCCCN(C(Cc3c(C)n[nH]c3)=O)C2)cccn2cncc12 C1(C2CCN(C(=O)CC3CCCC3)C2)(NC(CN(C(C(C)C)=O)C)=O)CC1 c1(CC(=O)NC(C2N(C(c3c(OC)ccs3)=O)CCCC2)C)c(C)nn(C)c1C Cc1csc2ncnc(NC3CC4CN(C(c5occc5C(C)C)=O)CC34)c12 N1(C(C2=NOC(CNC(c3cc(SC)oc3)=O)C2)=O)CC(O)CC(C)(C)C1 N1(C(CSCCC)=O)CCC(C)(C)CC1C(N1CCC(CC(=O)OC)C1)=O c1(CNC(c2cnc(SC)n2C)=O)cc(O)nc(CNC(C2CCOC2C)=O)n1 c1(CC(=O)NC2CC(N(C(C(CC3CCC3)OC)=O)C)C2)cc(F)ccc1C CCCCC(C(=O)Nc1csc(C)c1)NC(=O)CCCOCCC C1(c2n(CCOCC)nnn2)(Nc2ccc(C)c(Cl)c2)CCC=CCC1 CC1CCN(C(c2cc(C(F)(F)F)n(C)n2)=O)CC1NC(C1(C(N)=O)CCC1)=O C1(C)(CNC(C=C(C)C(C)C)=O)CCCN(C(=O)C2=NOC(C(C)(C)C)C2)C1 C1(C(=O)NCC)CCC(C)N1N1CC(OCCC=O)(CO)C1.C1(O)CC1 c1(C(=O)NCC2N(C(c3cnc(C(C)(C)CF)o3)=O)CCC2)cccc(=O)n1O C(=O)(C1CCc2cc(F)ccc21)N1C2(CNC(CCOCCOC)=O)CC(C1)C2 N1(C(=O)CCOC2CC2)CCC2CC2(C(N2CCc3c[nH]nc3C2)=O)CC1 N1(C(C2(C)N(C(c3cc(C)ncn3)=O)CC=C2)=O)CC2CC1C(F)(F)C2 C(=O)(C(F)(F)C(F)(F)F)NC1CCN(C(C23CCCC2C3(F)F)=O)C1 NC1CN(C(c2cc3ccsc3[nH]2)=O)C2(CCCOC2)C1 C(=O)(C(C(C)C)ONC(c1cn(C2CC2)cc1C)=O)NC(COC)(C)CO Cc1csc(C)c1C(N1CCOC(C2CN(C(=O)CCCCN(C)C)C2)C1)=O c1(CNC(C2CCC2NC(C2CCCN(C(C)=O)C2)=O)=O)cccc(F)c1O C1(C(=O)NCCCCCC=C)CC12CCN(C(=O)Cc1cccs1)CC2 C=CC(CCC)CC(=O)NC1(CCNC(c2cnccc2Cl)=O)CCOCC1 Cc1ccc(F)c(C(N2CC3CC3(NC(=O)C=Cc3cocn3)C2)=O)c1F CC1=NOC(C)(C(=O)NC2CCN(C(C3OCCC3C)=O)C2)C1 C1(CC)CN(C(=O)CCCOC(C)C)CC1C(=O)NCC(C)(O)CO c1(CCC(=O)NC23CC2CN(C(c2ccc(Cl)cc2)=O)C3)cccnc1Br C1(C(=O)N(C(C)CN(C(=O)CSC2CCCCO2)C)C)(NC(C)=O)CCCCC1 c1(C(N2CCCC(NC(C(CCC)CC)=O)CC2)=O)ccc2c[nH]nc2c1 C1(NC(C2(CNC(CCC(=O)NCC)=O)CC2)=O)CN(C)CC1(C)C c1(NCc2c(CC)nn(C)c2)[nH]c(=NCC2CC(C)(C)CO2)nc2sccc12 Cc1[nH][nH]c(=Nc2ccccc2)c1C(=O)Nc1ccc2c(c1)C(O)CCC2 C1(OCC)CCCC(C(=O)N(C)CCNC(=O)COCCCN(C)C)CC1 C1(C(=O)NCC2(CO)CCN(C(C3CCSC3)=O)C2)CCn2ccnc2C1 C(=O)(C(C)(C)CC(C)C)NCC1CN(C(COC)=O)CC(C)C1 C=CCC(CC(C)C)C(=O)NCCN(C(=O)CSc1ccc(NC(C)=O)cc1)C C1(C(N(C)CCNC(=O)C(c2ccc(Cl)cn2)(F)F)=O)CC12CCCCC2 O=C(CCC(=O)c1ccccc1)NC1(CCCNC(c2ccc(=O)oc2)=O)CC1 C#Cc1ccc(C(=O)NC(C)C=CC(N2CCC(C(C)CC)CC2)=O)nc1 c1(CN2CCC(NC(Cc3c(OC)ccc(Br)c3)=O)C2)cc(F)c(F)cc1Br c1(C(NCCNC(CCSCC)=O)=O)ccccc1.c1(C2CC2)ccccc1 c1(C(=O)NCC(C2CCN(C(=O)CCC(F)F)CC2)F)nccc2ncccc12 N1(C(c2c(CC)nn(C)c2)=O)CCCC(O)(CNC(=O)C2=C(Cl)CCCC2)CC1 S(=O)(=O)(c1ccc(NCC(C)(C)OC)c2cnccc12)NCCNC(=O)NC C1(NC(c2c(CCC)nsc2N)=O)CN(C(=O)CSS(C)(=O)=O)CC1C1CC1 C(=O)(C(C)(CC)CCC)NCC1(F)CCC(NC(c2c(OCC)oc(C)n2)=O)C1 C(=O)(CCCC(=O)N(C1CCCCC1N(C(=O)CNC(=O)C(C)(C)C)C)C)OC n1(CCNC(C2(CC)CC2)=O)cc(C(=O)NCCCOC2CC2)nn1 c1(NC(C)=O)cccc(C(=O)NCC(O)CCNC(=O)C=Cc2cncn2C)c1 Cc1ccc(C(N2CC=CC(NC(=O)Cc3ccc(O)nc3)C2)=O)cc1F CC1CC(NC(=O)C=C2CC2)CN1C(c1ccc(N2N=C(C)CC2=O)cc1)=O c1(C2CCCC(NCC(c3ccc4c(c3)CCC4)(C)C)C2)cc(F)c(F)c(F)c1 C1(C(N(CCCC(C)C)C)=O)N(C(=O)C(N2CCOC2=O)C)CC12CCCC2 CCCCC(C(=O)NC(C)CCC(=O)N1CCCC1C(O)CO)NC(N)=O C(C)(CCC(=O)NCC1(O)CC(NC(c2coc(C#N)c2)=O)C1)SC c1(CNC(C2N(C(c3c(CC)nccc3)=O)CC(OC)C2)=O)cc(C)cnc1O C1(OC)CC2(C1)CC(C(=O)CC1CC(c3nnnn3C3COC3)(N)C1)C2.OC c1(CN=[N+]=[N-])ccc2c(c1)CN(Cc1ncc(Br)cc1Cl)C2 N1(C(C(CCN(C)C)O)=O)CCCCCC(NC(C2COC2)=O)C1 N1(C(c2[nH]cc(C(N)=O)c2)=O)CCCCC1C1CCCN1c1nnc(C2CC2)o1 c1(C(N2CCCC(C(C)NC(=O)C(F)=CC3CC3)C2)=O)ccncc1N=[N+]=[N-] N1(C(C(C)C2CC2)C(=O)NCC2CCOCC2)CC=C(C(N)=O)CC1 C(N=c1[nH]c(C)ncc1F)C12CC(CNC(CCOCCOC)=O)(OC1)C2 C1(F)(CNC(C(CCC)OC)=O)CCCN(C(C2CNC(=O)C2)=O)CC1 Cc1nc(C)c(CC(=O)NC2CN(C(c3cn(CC4CC4)nn3)=O)CC2C)s1 C1(CC(=O)NCC(=O)Nc2cc[nH]c2)(NC(COC(C)(C)C)=O)CCC1 C1(NC(CCCCC)=O)CN(C(=O)CN(C)Cc2ccccc2)C2(CCOC2)C1 C1(OC(C)C(=O)NCC2CC2NC(=O)C=CC2CCC2)CCCCCC1 Cc1ccc2c(C(N3CCC(NC(=O)CC45CC(C4)C5)C3C(C)C)=O)n[nH]c2c1 Cc1cccc(C2CCCN2CC2(C)CCCNC2)c1 N1(C(C2(SCC)CC2)=O)CC2CN(C(c3cncnc3CC)=O)CCC2(CO)C1 c1(C(=O)NCC(C)CN(C)C(C2(C#N)CC2C(F)(F)F)=O)ccc(Cl)[nH]1 c1(C(N(CCN(C(C2C(C(C)C)(CC)C2)=O)C)C)=O)cc2ccncc2cc1F c1(C(=O)NCC(CNC(CNC(=O)NC)=O)O)cc2c(s1)CN(C)CC2 C=C(C)C(C)(C)C(=O)NCCCN(C(=O)C(=O)NCC)C1CCCC1 CC1CN(C(C2CC2F)=O)CCN1C(c1cn(CCCF)nn1)=O c1(C(=O)NC23C(CN(C(C4C(=C)C4)=O)C2)C3)cc(F)c(F)c(N)c1Cl C1(CNC(C2CN(C)C(=O)C2)=O)CN(C(c2cc3cscc3s2)=O)CCN1C N#Cc1cccc2c1CCCN2C(=O)NNC(=O)C1CC1c1ccc([N+](=O)[O-])cc1 Nc1ccc(C(=O)NC2CCN(C(c3cc(C(F)F)ncn3)=O)C2)c(Cl)c1 Cc1noc(Cl)c1CC(=O)NC1(CO)CCN(C(=O)Cc2nc[nH]n2)C1 c1(SC)ccc(N2CC(C(N3CCOC(c4cnn(C)c4)C3)=O)CC2=O)cc1 N1(CCNC2(c3n(CCCSCC)nnn3)CCOC2C)C(=O)COCC1=O n1(CC)nc(C(=O)NN2CCC2Cc2cn(C3(C(=O)O)CC3)nn2)cc1O Cc1cccc2[nH]cc(CC(N3CC(C)CC(C)C3C(=O)O)=O)c12 c1(C(N2CCC(O)(CCNC(CCOC)=O)C2)=O)nc(O)nc(O)c1N C(=O)(C(CCCCC)C(C)C)NCCCC1(NC(CN(CC#C)C(C)=O)=O)CC1 c1(C(N2CC(NC(C(CC)NC(c3ccco3)=O)=O)C2)=O)cc(C)nn1C(F)F N=c1[nH]c(Cl)c([N+](=O)[O-])c(=NCC(O)CNC(c2cc3ccccn3n2)=O)[nH]1 C1(NC(=O)Cn2cc(-c3ccccc3)cn2)CNCCC1CO C1(C(=O)NCC(c2ccc(O)cc2)O)C2CCS(=O)(=O)C12 N1(C(c2nc(Br)ccc2F)C(=O)NCC2CCCO2)CCn2ncnc2C1 c1(CCNC(=O)NCC2(C)CC=CCC2)c[nH]c2ccccc12 C(=O)(C1CNC(=O)c2ccccc21)N1CC2C(NC(=O)CN3CC4CC4C3)C2C1 C1(NC(CC(C)(C)F)=O)CC2CCC(C1F)N2C(=O)Cn1cc(P(C)(C)=O)cn1 C1(CC(=O)NC(CNC(C(C)N(C)C)=O)(C)CO)CCC(C)(C)CC1 C1(=CC(=O)NC2C(NC(C(CCC)OC)=O)CCC2)CN2CCC1CC2 C1(C(=O)NC23CC(NC(c4nn(CC)c(O)c4)=O)(C2)C3)CC12CCCCC2 N1(C(C2C(C)CCO2)=O)CC(C)(C)CC1CNC(=O)Cn1cc(C2CC2)cn1 CC1COCC(CNCc2cccc(-n3ccnc3)c2)O1 N1(C(c2c(C)ncs2)=O)CCN(C(c2ccc3nc(O)[nH]c3c2)=O)C(C)CC1C CC(O)C(C(=O)N(C)CC1CCN(C(c2ccc(C#N)o2)=O)C1)N(C)C N1(C(C2C(CC(C)(C)C)C2)=O)CC2CC(C1)CN(C(c1c[nH]nc1C1CC1)=O)C2 N(C1CCC(c2ccc(Cl)c(Cl)c2)c2ccccc21)C(C)CN1CCCNC1=O c1(C(N2CCC(c3cn(-c4cccnc4)nn3)C2)=O)ccc(-n2cncn2)nc1 c1(C(=O)NCC(COC)NC(C2SCCCS2)=O)cc(OC)n[nH]1 C(C(CNC(c1ccc(O)cc1Cl)=O)C(F)(F)F)NC(C(C)(C)OC)=O CCCC(O)CC(=O)NC1CC(N(C(=O)Cc2c(C)nn(C)c2C)C)C1 CCCC(C)C(=O)N1CC(NC(=O)CCc2nc(O)n[nH]2)C(n2ccnn2)C1 CCC(C)CCCCC(=O)N1CCCC(N(C)C(c2ccc(C3CC3)cc2)=O)C1 C1(NC(c2cccc(SC)c2)=O)COCCN(C(C2CC3(C2)CC(F)C3)=O)C1 c1(CN2CC3C(NC(CC(C)C)=O)C3C2)cc(F)c(F)cc1Cl CCCC(CC(C)C)C(=O)N1CCC(C(F)CNC(=O)CCOC(C)C)CC1 C1(CNC(c2c(OC)ccnc2)=O)C(C)CCCN1C(C1CC(=C2CCC2)C1)=O N1(C(C(CC)C(C)O)=O)CCC(N=c2[nH]c(C3(OC)CCCC3)nc(=N)[nH]2)CC1 N1(C(C2(CNC(=O)CCCn3cccn3)CC=CC2)=O)CCCCC1CCCO C1(NC(COCCC=C)=O)CC(O)CN(C(c2ccn(CCC)n2)=O)C1 C(=O)(CN=c1nc2sccc2c(NCC2CCOC(C)C2)[nH]1)N(C)CC N1(C(COCCC=C)=O)CCCN(C(c2cc(C)cc(F)c2)=O)CCC1 c1(C(=O)NCC2(NC(C3CC(C)(CC)C3)=O)CCCCC2)sccc1S(C)(=O)=O N(C(=NCC(c1ccco1)OC)NC1CCC1)CC(CC)(C)COC c1(C(=O)NC(C)CCCNC(c2c[nH]nc2C2CCOC2)=O)ccnc(S)c1 CON1CCC(C(=O)N(C)CCNC(C2CCC(COC)O2)=O)CC1 C(=O)(C(C(C)C)n1cc(C)cn1)N(C1CC(CNC(COC)=O)C1)CC(C)(C)C Cc1ccnc(Cl)c1C(=O)N(C(C)CNC(=O)CCCC(N)=O)C C=CC(C)(C)C(=O)N1CCC(CCCNC(=O)Cc2ccccc2C)CC1 c1(C(N(CC(C)NC(c2c(C)nn(C(C)C)c2C)=O)C)=O)ccc2cnoc2c1 C(=O)(CC1=CCN(C(C2(C)CCC(C)C2)=O)CC1)Nc1ccc(C)nc1O c1(CNC(CC=CCNC(C(C)c2cc[nH]n2)=O)=O)cc(O)ns1 c1(C(=O)NC(C(C)NC(C(C)OCCOCC)=O)CO)cc(CC)nn1C c1(C(C(N2CC(c3cn(CC(C)(C)C)nn3)(C)C2)=O)(C)C)cccc(Cl)c1 C1(NC(c2c(Cl)cn(C)n2)=O)CC2CCC(C1F)N2C(c1cc(C2CC2)on1)=O C1(C(=O)NCC(C)NC(C(C(C)C)NS(C)(=O)=O)=O)CCc2ccccc2O1 C(=O)(CCCS(C)(=O)=O)NC(CNC(c1cnc(C(C)C)o1)=O)(C)C(C)C N1(CCC#C)CCC(C(N2CC(O)(CCNC(=O)C(O)CC3CC3)C2)=O)CC1 N1(C(C(CC)C)=O)CCC(N(C)C(c2ccc(C(C3CC3)OC)nc2)=O)CC1 CCC(O)C(C)C(=O)NCC(C)N(C)C(c1cc(Br)c(C)s1)=O Cc1nc(C2CC2)oc1C(=O)NCCCNC(=O)C(N1CCNC1=O)C C1(O)(CCNC(C2(CC)CCCCC2)=O)CCCN(C(c2ccc(O)nn2)=O)C1 C1(NC(C2(S(C)(=O)=O)CC2)=O)CC2(C1)CC(NC(C1(C)CCNC1=O)=O)C2 C(=O)(CC(C)(C)O)NCCc1c(C(N(CCS(C)(=O)=O)C)=O)c[nH]n1 C1(CNC(C(C)N(C(C)=O)C)=O)(OC)CCN(C(=O)C=C(C)Cl)C1 N1(C(C2CC(NC(CC3CC(=C)C3)=O)C2)=O)CC(CO)C2(CCC2)C1 c1(C(c2n(C)nnn2)NCCC2CC(C)(C)CCO2)sc([N+](=O)[O-])cc1Cl C(=O)(CCCC(OC)OC)NCc1ccc(CNC(C(CCC)=CCC)=O)cc1 CC1(C)CCCN(C(=O)OC(C)(C)C)C1C(=O)Nc1ccc(O)cc1C#N C1(C(N(C)CC2CCCC3CC23)=O)CCN(C(=O)CC2CCCN2C)CC1(C)C CC1=C(C(=O)NC2CCN(C(=O)C=Cc3ccco3)C2)C(C)n2ncnc2N1C CCC(CCC(=O)N1CCCC1C1(O)CN(C(c2cc(C(C)C)no2)=O)C1)OC c1(C(N2CC(CC(C)NC(C(COC)OC)=O)C2)=O)cc2sc([N+](=O)[O-])cc2[nH]1 N1(C(C(C(CC)C)NC)=O)CC2COCC(C1)C2NC(=O)Cn1nc(C)cc1C Cc1ccc2c(c1)CC(C(N1C3CCC1CC(N(C(=O)C(F)F)C)C3)=O)S2 Cc1cccc(C(=O)NC(C2CCCCC2)C(=O)NCCC(C)C)n1 c1(C(N2C(C(NOCC(=O)N(C)C)=O)C=CCC2)=O)ccc2c[nH]nc2c1 c1(C(=O)NC(CNC(CNC(C(CC)C)=O)=O)C(C)C)ccc2oc(O)nc2c1 c1(C(C)(C)C)cccc(C(N2CC(NC(c3sccc3Cl)=O)C3(CC3)C2)=O)c1N N#Cc1ccc(CC(N2CCC3(NC(c4ccc(Cl)[nH]4)=O)CC3C2)=O)cc1 Cc1cc(C(N2CC3CC(NC(=O)CC(C)(C)O)CC2C3)=O)c(F)cc1F N1(C(C(CN(C)C)O)=O)CCCC(NC(C2COCC2(C)C)=O)C1 C1(CNC(=O)CCc2ccsc2)C2CN(C(c3ccn(C4CCCC4)n3)=O)CC12 C1(C(=O)NC(CNC(c2n(C=C)ncc2)=O)CCC)COc2cc(Cl)ccc2C1 c1(C(=O)NCCNC(C2N(C(CCCC)=O)CSC2)=O)cnc2c(c1)COCC2 Nc1cc(C(N2CC3CC2C3NC(c2cnsc2)=O)=O)cc(O)c1 c1(C(N2CCCC(C3CCCCN3C(=O)CCCCO)C2)=O)cnc(F)c(F)c1 c1(CNC(C2CCCC2O)C)ccc2nc(N(C)C)[nH]c2c1 C1(NC(COCCOC)=O)CN(C(c2cc(OC)c(F)c(F)c2)=O)CC2(CC2)C1 C(CC(C)C(=O)NC(C)C(CO)NC(c1csc(Br)c1C)=O)OC CCCC(F)(F)C(=O)NCC1CCCN1C(=O)COCC(C)(C)C n1(CCCC)nc(C(=O)NC2(CCNC(C3CC=C(C)CC3)=O)CC2)ccc1=O C1(C(=O)NCC2(F)CN(C(Cc3c(C)con3)=O)C2)C(C)(C)C1(C)C c1(C(=O)OC)c(O)nc2c(OC)cccc2c1NC1CCCCCC1F C1(CNC(CC2ON=C(CC)C2)=O)CC(C)(C)CN1C(c1cccc(Cl)c1F)=O C1(COC)CN(C(=O)C(C)C2CC2)CCN1C(=O)CCc1cscn1 N1(C(C2C(=C)C2)=O)CC2CCN(C(=O)C=Cc3cccc(F)c3Cl)CC(C2)C1 c1(C(N(CC(C)O)CCNC(=O)COc2ccccc2)=O)cc2c[nH]nc2s1 C(c1cncc(O)c1)=CC(=O)NC1CCC(N(C(C=CC(=O)OCC)=O)C)C1 N1(C(C(CCC=C)(C)C)=O)CC2(CCN(C(=O)C(CO)C(F)(F)F)CC2)C1 N1(C(C(SC)SC)=O)CCCCC1CCC(=O)NCC(=O)N(C)O c1(C(=O)NCC2C(NC(c3snc(O)c3Cl)=O)C2)cc2ccc(O)cc2[nH]1 C(CCCCC(=O)NCC(c1cnn(C)c1)O)N(C(=O)C(O)c1ccco1)C Cc1cncc(C(N2CCCC(C(C)NC(=O)Cn3nnnc3C)C2)=O)c1Cl CN1CCC(C)(C(=O)NCC2CC3CC3N2C(c2cnn(C(C)(C)C)c2)=O)C1=O c1(OC)ccc(C2=NOC(C(=O)NC34CCC(C)(CC3)CO4)C2)cc1F C1(CNC(c2c(C)nc[nH]2)=O)CN(C)CCN1C(C1CC(OC2CC2)C1)=O C1(CNC(C2CCCCS2)=O)CC2CCC1N(C(C1CSCCS1)=O)C2 Cc1onc(CO)c1C(=O)NC1CCCC(NC(C2CC2c2ccccc2)=O)C1 CN(C)NC(=O)CCC(=O)N1CC(N(C(=O)C#CC2CCCOC2)C)C2(CC2)C1 C1(c2ccccc2)(C(=O)NCCN(C(=O)C(O)CN(C)C)CCOC)CC1(C)C N1(Cc2nc(-c3ccc(C)cc3)oc2)CCC(SCC2CCCCCC2)C(C)C1 C1(C(=O)NC2CCN(c3ccccn3)CC2)CC2CCC(C1)S2(=O)=O c1(NC(C(C2CC3CC3N2C(=O)NCCCl)C)=O)cccc(C(N)=O)c1 N#Cc1cnc(C(=O)NCCCNC2(c3ccc(C(F)(F)F)cn3)CC2)c(F)c1 CC1(C)CCCC(C(N2CCCC(CNC(c3n[nH]cc3C(F)F)=O)CC2)=O)C1 CC1CN(C(=O)CCOCC2CC2)CCCN1C(c1cscc1F)=O C#Cc1cc(F)c(C(=O)NCCC(C)(C)CNC(=O)CC2CCCCO2)c(F)c1 c1(C(=O)NC2C(CC)N(C(c3nc(C)c(C)s3)=O)CC2)cc2occc2n1C c1(C2(C(N3CCC(C(C)C)C3)=O)CCC2)ccc(Br)cn1 c1(C(=O)NC2C(CNC(C3(CCC=C)CCC3)=O)C2)cc(Cl)ncc1OC N1(C(CC23CC(C)(OC2)C3)=O)CCCC2CN(C(C3OC(C)CC3C)=O)CC12 Cc1cncc(C(=O)NCC2(NC(=O)Cc3ccsc3C)CCCC2)c1 c1(C(N2C(C)CC(CNC(=O)Cn3ccccc3=O)C2)=O)ccc(Cl)cc1O C1(C)(CNC(CCOCCC)=O)CCC(NC(=O)CCCCOC)C1 Cc1n[nH]c(C)c1CC(C)C(=O)NC1(CNC(C2CCC(C(N)=O)N2C)=O)CC1 N1(C(C)=O)CCCCC1CC(=O)N(CCNC(C1(C)CC(C)=NO1)=O)C(C)C C1(C(N2C3CN(C(c4cc(Cl)no4)=O)C(C3)C2)=O)COc2cc(Cl)ccc2C1 CCCS(=O)(=O)C(C)C(=O)N1CCC2(CCN(C(c3csc(COC)n3)=O)C2)C1 Cc1cc(C(=O)NC(C)(CNC(C2CCNC2=O)=O)CO)c2nccn2c1 N1(C(C(C)Cn2ccnc2)=O)CC2=CC2=NNC=CCC1C(=O)O CC(C)C(CCN(C)C(c1cccc(C(N)=O)c1)=O)NC(c1cccc(F)n1)=O c1(N2CCC(NC(C(C)(C3CC3)OC)=O)CC2C)nnc2c(c1C#N)CCCC2 C1(C(=O)NCc2oc(C)c(C(=O)N(C)CC3(O)CCOC3)n2)CCC=CCCC1 C1(NC(c2ccsc2)=O)CCN(C(=O)C=Cc2ncco2)C1c1ccccc1 C#CCC(C(=O)OCC)NC(=O)CC1(N(C(=O)CSCCOC)C)CC1 N1(C(=O)C(O)Cc2ccccc2)CCN(C(=O)Cc2cccc(Br)c2)CC1 C1(C(=O)Nc2c(C)cccc2O)C2CC(O)C(C2)N1C(C1(C)CCSCC1)=O C1(NC(c2ccc(C)nc2N)=O)CS(=O)(=O)CC1NC(=O)CNC(=O)CN(C)C N1(C(C(=O)N(C)Cc2c(CC)noc2)C)C(=O)NC2(CCCC2)C1=O C12(CNC(C(CC#C)C3CC3)=O)CCC1CN(C(c1cc(C)nc(C)n1)=O)C2 C(C(C)(C)CNC(=O)NCC1(C)CC1(F)F)OC c1(OC)cc(OC)c(-c2nccn2C(C)C)cc1OC(C)C.C1=CC=C(C)CC1 C(C1CCN(C(=O)Cc2cnns2)CC1)=CC(=O)NCC(C)(F)CCCO c1(C(=O)NC2(C#C)CC2)sccc1CNC(C1CCCCO1)=O C(=O)(C1CC(=O)c2c(F)cccc21)NCCC1CN(C(CC=C)=O)C1 c1(C(N(C2CCN(C(c3ccnc(C)c3N)=O)C2)CC)=O)cc(F)c(F)cc1F C(CCCCS(C)(=O)=O)NC(C(C(C)C)(C)C)c1nnnn1CC1CCCO1 Cc1cc[nH]c(=N)c1C(=O)NCC12CC(NC(c3ccc(Br)o3)=O)(CO1)C2 Cc1ncsc1C(=O)NCCN(C(=O)CC1(NC(C2(C)CCC2)=O)CC1)C(C)C C1(N(C)C(c2csnn2)=O)CN(C(=O)CCC(=O)c2ccc(Cl)s2)CC1F N1(C(c2cc(C)c(C)s2)=O)CCC2C(CCN2C(=O)COc2ccccc2)C1 N1(C(Cc2ccc(OC)cc2)=O)CCCN(C(=O)C=CC(=O)N(C)C)C(CO)C1 C1(CCCNC(CCC)=O)CN(C(C2CC2CN(C)C)=O)CCO1 c1(NC(C(C)OC(c2nc(C(C)C)oc2)=O)=O)cccc(C#N)c1 C=C1CC2CCCC(C1)N2C(C1CCCCC1(C)NC(c1sc(O)nc1C)=O)=O c1(COCC)nnc2n1CCN(C(=O)NC(C)(CC(F)(F)F)c1ccccc1)C2 C1(CC(=O)NCC2(CSC)CC2)CCCC(NC(=O)COCC2CCCO2)C1 C(=O)(C1=CCCC1(C)C)N1CC2C(CNC(C3CCN(C(=O)NCC)C3)=O)C2C1 c1(NC(CC2CC(NCc3scc(C)n3)C2)=O)cc(Cl)cc(Br)c1C N1(C(Cc2n(C)ccn2)=O)CCN(C(c2ccc(C#N)[nH]2)=O)C(CC(F)F)C1 c1(C(N2CCCC(C(=O)NC(COC)C)CC2)=O)cc([N+](=O)[O-])ccn1 c1(CC(N2CC(NC(CCCOC)=O)C(C)C2)=O)ccc(Br)cc1[N+](=O)[O-] c1(OC)ncc(C=CC(=O)NC2CCC2NC(=O)C(C(C)C)NC(N)=O)cn1 c1(C(=O)NCCC(C)(C)NC(C2CC3CC2C2CC32)=O)cnn2c1OCCC2 c1(C(=O)NCC(C)(C2CC2)NC(C(CC)OCC)=O)c(C)nn(CC(C)C)c1Cl N1(C(C2C3COCC23)=O)CCN(C(C2CC2F)=O)c2ccc(Cl)cc2C1 N1(C(C(C(C)CC)N(C(COCCC#C)=O)C)=O)CCC(C)C2(CCC2)C1 C1(NC(=O)NCC(c2ccc(C)o2)N2CCOCC2)CC2(CCC2)C1O Cc1[nH]c2c(C(=O)N(CCCCNC(C3CCC(C)O3)=O)C)cccc2c1C c1(C(N2CCC(C)(NC(c3c(CC)scn3)=O)C2)=O)cnc2c(C)cnn2c1 CN1CCCCC1C(=O)NCC(c1ccccc1F)NC(c1cc(Br)no1)=O c1(CC(N2CC(NC(CCCNC(=O)OCC)=O)C(C)C2)=O)ccc(F)c(F)c1 c1(C(N2CCC(N(C)C(c3cnc(C4CC4)s3)=O)C2)=O)occ2c1CCOC2 C1(NC(C(=Cc2cccs2)C)=O)CN(C(=O)CCc2nccn2C)CC2CC12 c1(C(=O)NCC2CCCCCN2C(=O)Cc2ncsc2Cl)csc2c1CCCC2 c1(C(N(C)CCC2CCCCN2C(C2CCC3CC23)=O)=O)cc[nH]c(=N)c1Cl c1(NC(c2c(OC)nccc2)C)[nH]c(=NC2CC=C(C)CC2)nc2sccc12 C(CC(C(C)(C)C)NC(c1cc(C(F)(F)F)ns1)=O)N(C(=O)C1=CCOC1)C C(C(C)(O)CC(=O)NC(C1CCN(C(=O)Cc2coc(C)n2)CC1)(C)C)OC CC1CC(NC(c2csc(C(F)F)n2)=O)CCN1C(=O)C=CC1CCCCCC1 O=S(=O)(c1ccc(-n2cccc2)nc1)N(C1(c2ccccc2)CCC1)CCCO c1(SC)cc(C(=O)NCC2CC(CNC(=O)CSC(C)C)CO2)ccc1F CCC(CC(=O)NC(CO)CCCCNC(c1c(C)ccc(Cl)c1N)=O)C(F)F C(CC(=O)NCc1cc(O)ccc1F)(C(F)F)NC(c1nc(OCC)oc1)=O N1(c2n(C3C4(CCOCC4)C3)nnn2)CCCC12CCOC2 C1(C(F)F)(NC(CN(C)C)=O)CC(NC(=O)C(=O)NC2CC2)C1 c1(NC(C2(c3ccccc3Cl)CCC2)=O)cc(Br)cc([N+](=O)[O-])c1 N1(C(c2[nH]cc(CC(C)C)c2C)=O)CCN(C(=O)C2CC2)CC1(C)C N1(C(C(CC)N(C(=O)C=CCO)C)=O)CCc2nncn2CC1 Cc1oc(C#N)cc1C(=O)N(CC(C)(C)CNC(c1ccc(O)nc1)=O)C C(c1ccc(F)c(F)c1)=C(C(=O)NC(CCNC(C1(CC)CCC1)=O)C)C C1(NC(CNC(N)=O)=O)CN(C(=O)Cc2ccc(C(N)=O)nc2)CCC1O CCC(C)C(O)C(=O)NCC1(F)CCN(C(c2ccc(-c3ccon3)cc2)=O)C1 C1(C(C)NC(c2n(CC=C)ccc2)=O)CCN(C(C2CCCCC2OC)=O)CC1 N1(C(C(CNC(C)=O)(C)C)=O)CC=C(C(=O)N2CCOCC(CO)C2)C1 c1(C(C)C)nc(NCCCN2CCN(C)CC2)cc(=NC2CC=CCC2)[nH]1 C=CCCCCC(=O)NC1(CC)CCCN(C(c2ccc(CC3CC3)s2)=O)C1 CCC(C(C)(F)F)NC(=O)COC1(C)CN(C(C2(COC)CCCO2)=O)C1 N1(C(c2ccc(OC)s2)=O)CCC(CNC(c2nnc(O)nc2O)=O)C12CC2 c1(C(N2CCC(CCC(=O)N(C(CO)C3CC3)C)C2)=O)ccc2cc[nH]c2n1 c1(C(=O)NC(CNC(c2cc(OC)n(C)n2)=O)(C)C(C)C)cc(O)nc(O)n1 Cc1onc(C2CC2)c1C(=O)NC1CN(C(C2(CF)CC2)=O)CC1C c1(OCC)cnc(N2CCC(N(C(=O)CCC3CCC3)C)CC2)nc1C C12(N(C(CCCCC)=O)c3ncc(Cl)cn3)CCC(CC1n1cc(C3CC3)nn1)C2 c1(NCc2cc(C(=O)OC)c(C)o2)ccnc(CO)c1C C1(NC(C2CC(=O)NC2)=O)CCC2(CC1)CN(C(C1(CCF)CC1)=O)C2 c1(SC)ccc(C=CC(=O)NCC2(O)CCN(C(C3CCCN3C(C)=O)=O)C2)s1 C(CC(C(=O)NC(C)(CNC(=O)CCc1ccccc1F)C1CC1)NC=O)SC c1(OC)c(Cl)cc(O)c(Cl)c1C(=O)NC1CCCC1NC(C1(COC)CCC1)=O C1(CNC(C(C2CCN(C(CCc3ccn(C)n3)=O)C2)(C)C)=O)CCC(=O)NC1 c1(C(C(F)(F)F)N2CCC(CNC(=O)Cc3ccccc3Cl)C2)ccc(Cl)cc1 C1(COC(=O)NCCCC)CCCCN1C(C1CCOC(C)C1)=O C1(C(N(C2CCN(C(C3C(=C)CC3)=O)C2)CC)=O)CC2(CC(=O)N2)C1 C(=O)(CC1=CCOCC1)N1CC(NC(c2cccnc2O)=O)CC(C)C1 C1(CC=C)(NC(=O)CCOC)CCCN(C(=O)CC2CC2C2CC2)C1 c1(NCCCNS(CC)(=O)=O)[nH]c(=NCC2(C)CCC(=O)N2)nc2c1cnn2C c1(C(N2CCC(C(CNC(CCOC)=O)F)CC2)=O)oc2ccccc2c1Cl Cc1ccc(F)c(C(=O)N(C2CN(C(C3CCCN3C3CCCC3)=O)C2)C)c1 c1(OCC)ccc(S(=O)(=O)NC2CCNC(=O)C2)cc1-c1ccc(C)cc1 C1(CNC(CN(c2ccccc2)C(C)=O)=O)C2CN(c3ncc(Cl)cn3)CC12 C1(NC(C(C(C)C)NC(C)=O)=O)CCC2CCN(C(c3ncnn3C)=O)C1C2 CC(C)CC(O)CNC(=O)C(=O)NCCNC(c1ccco1)C C1(CNC(=O)CCC2CCC2)CCN(c2nc(CC3CC3)ns2)C1 N1(C(CNC(c2c(C)ccn2C)=O)=O)CC2(CCC(O)CC2)C1 Cc1nc2c([nH]1)CN(C(=O)CN(C(=O)CCCC1CC1)C1CCC1)CC2 N1(C(Cc2ccn(C(C)C)n2)=O)CC2CC2(NC(c2cc(Br)cs2)=O)C1 c1(OC)c(C)cc(C(=O)Nc2cccn(CCn3cccn3)c2=O)cc1N N1(C(c2c(N)snn2)=O)C2CCC1CC(C(=O)NC1CCCC(C3CC3)C1)C2 c1(CC(N2CCC(C(C)NC(C3CCC(C(N)=O)O3)=O)C2)=O)ccc(F)cc1F C1(N(C(=O)CSCc2ccccc2)C)CN(C(c2ccsn2)=O)CC1(C)C C=CC(CCC)CC(=O)N1CC(OC)CC1CNC(=O)C=CC(=O)N(C)C N1(C(c2c(C)nccn2)=O)CC(NC(c2csc3cccnc23)=O)C(C2CC2)C1 C(=O)(CCCCC(N)=O)NCCCC(C)NC(c1cc(OC)c(O)cc1)=O n1(CCC#C)c(N(CCCn2ccnc2)C)nnc1-c1coc(=NC)[nH]1 O=C(CCCCn1ccnn1)NC1(CF)CCN(C(=O)CCn2cnnn2)C1 C(CC(C(C)C)NC(=O)C(C)NC(C)(C)CC)N(C(COCCC#C)=O)C C1(O)(CNC(CC2CCN(CC(C)C)C2)=O)CCN(C(=O)NC2CCCO2)CC1 C1(C(=O)NCC2(C)CCCN2C(C2CCCN2C=O)=O)Cc2ccc(F)cc2C1 C1(O)(CN(C)C(C2(C(F)F)CCCC2)=O)CCN(C(c2cnc(Cl)[nH]2)=O)C1 c1(NC(C)CCC2CCCO2)nc(N2CC3CCC(C2)C3(F)F)nc2sccc12 CCCCC(O)C(C)C(=O)NC1CN(C(=O)CC2CC(F)C(=O)N2)CC1SC C1(OC)(CNC(=NCC2(C)COCCO2)NCC(F)F)CCCSC1 CC1CN(C(C2CN(C)C2)=O)CC(C)N(C(c2ccc3sccc3c2)=O)C1 C1(CNC(C2CC=CCC2)=O)CC2COCC2N1C(c1occ2c1CCC2)=O c1(C(=O)NC2(CNC(C(CCSC)O)=O)CCCC2)ccc2snnc2c1 CCCC(CC1CCCC1)C(=O)NC(C)CN(C)C(c1c[nH]ccc1=N)=O C(=O)(C(F)CC(C)C)N1CCC(N(C(=O)Cc2cc(C3CC3)on2)CC#C)CC1 C1CCCN1C(=O)C(C)OCCC(C)C.CC(C)CN(CC(N)=O)C=O N1(C(CC(CC)(F)F)=O)CCC2CN(C(c3cc(C4CC4)ncn3)=O)CCC2C1 c1(C(=O)NC(CC)CNC(c2ccnc(SC)c2)=O)cnc2nccn2c1 C1(C(N2CC(CNC(C(C(C)OC)N(C)C)=O)C2)=O)CC2(CCC(F)(F)CC2)C1 C1(OCC(N2CC(=C(CNC(C3C(OC)C3)=O)F)C2)=O)CCCCC1C N1(C(C(C)c2ccsc2)=O)CC2CC2(C(=O)NCc2nnc(C3CC3)o2)C1 C(c1ccc(OC)cc1C)=CC(N1CCC(c2cccc(OC)c2)C1)=O CCCCC(CC(=O)N1CC(C)(C)C2COCC12)NC(C1OCCC1C)=O C1(C(C)C)CCCC(NC(=O)CN(c2ccccc2)CC(=O)O)CC1 C1(CC=C)(CNC(c2csc(CNC(C3COC(=O)N3)=O)c2)=O)CCCC1 N1(C(C=CC=CC)=O)CCC2CCN(C(c3cc(F)c(O)c(F)c3)=O)CC2C1 c1(N2CCCC(CC)(CC)C2)nc(NCC(C(C)(C)C)OC)c2cnn(C)c2n1 CC1CCc2c(sc(NC(=O)C(=O)NCC3CCN(C)C(C)C3)c2C#N)C1 CN1C(=O)NCC1C(N1CCCC1(C)CNC(=O)CCN(C)CCO)=O C1(NC(c2cn(CC(F)(F)F)nn2)=O)CCN(C(c2cccs2)=O)C1 c1(CNC2(c3n(C(CC)C)nnn3)CCN(C)CC2)ccc(S(C)=O)cc1 O=C(CCCCc1ccccc1O)NC1CCC(C2CC2)C1.C12(CC1)C(=O)NC2 c1(C(N2C(C#C)COCC2)=O)ccc(S(=O)(=O)NC)nc1 CC1(CC(N2CCC(O)(CNC(c3cc(C(N)=O)cs3)=O)C2)=O)SCCCS1 c1(N2CCC(OC)(CO)C2)ccc(S(=O)(=O)N2CCS(=O)(=O)CC(C)C2)cc1Cl C(=O)(C(C(C)C)SC)N1CC(NC(c2c(CC)c[nH]n2)=O)C1 n1(CC(N2CC(C(C)NC(C(CSC)C)=O)C2)=O)ncc(C#N)c1N C(=O)(CC(CC)C(F)F)NC1CC(COCC)CN1C(=O)CCc1nccn1C CCCCCCC(=O)NC(CNC(c1nc(C)sc1Br)=O)(CC)CC c1(C(N2CC(O)(CCNC(C=COCC)=O)C2)=O)[nH]c(Cl)c(Cl)c1Br CN1CCCCC1Cc1nc(Cn2cncn2)nn1-c1ccccc1 C1(NC(C(c2cc(C)cc(C)c2)C)=O)CCC2CCN(C(=O)CC3CC34CC4)C12 c1(C(N2CC(CCNC(C=NOC)=O)S(=O)(=O)CC2)=O)cc(F)c(F)c(C#N)c1 N1(C(c2c(CC)nccc2)=O)CCC2(NC(c3cnnn3C)=O)CC2C1 N1(C(c2cc(OC)c(C(F)(F)F)cc2)=O)CCCN(C(C2CCCO2)=O)CCC1 C(=O)(CC(O)CC(C)(C)C)N(CC(C)O)Cc1cccnc1.C1(=O)CN1 Cc1oc2ncnc(O)c2c1C(=O)NC1CCCC(CNC(=O)CP(C)(C)=O)C1 c1(NC(=O)NC(c2ccccc2OC)CC(=O)OCC)ccc(C)c(CN)c1 N1(CC(=O)NCCC2CC(NC(CSc3nc(C)[nH]n3)=O)C2)CCCS1(=O)=O C1(NC(=O)N(Cc2ccccc2)Cc2cccs2)CCN(CC2CC2)C2(CCC2)C1 CC(CC(=O)N(CCCOCCNC(c1nnc(O)cc1O)=O)C)CC(F)(F)F N1(C(CC(CC)(C)C)=O)CCC(N=[N+]=[N-])(C(N2CC3(CCC3O)C2)=O)C1 CC#CC1CCN(C(=O)Nc2c(C)ncnc2C)C1 CC1(C)CC(C(N2CC(CO)(NC(c3cnns3)=O)C2)=O)CO1 Cc1nn(C)c(C)c1CC(=O)NC1CN(C(c2cccc(F)c2O)=O)CCC1O C1(C(=O)NC(C)(C)C)CCCC(NC(=O)Cc2ccccc2F)C1 C(=O)(CC(C)C(C)C)N(CCOc1cccc(NC(c2scc(CC)c2)=O)c1)C c1(-c2cn(CC3OCCN(C(CN(C)C4CC4)=O)C3)nn2)cccc2o[nH]c(=N)c12 c1(C(=O)NC2(C(=O)Nc3cc(C)c(O)cc3)CCOCC2)ccc2nccn2c1 CC(CC(C)NC(=O)C(c1ccc(Cl)s1)C)NC(=O)CN(C)C c1(C(c2nnnn2CCCSCC)NCCCCOCC)coc(C)n1 N1(C(c2ccc(OCCC)cc2)=O)CC=C(CNC(C2CC3CCC2O3)=O)CC1 c1(C(C(=O)NCCC(CC)O)N(C)C)cccc(Br)c1 C(CCCC(=O)N1CCCC1C1(O)CN(C(C2CC=CCC2C)=O)C1)OC N1(C(c2c(C)ccs2)=O)CCC2CCC(C1)N2C(c1cn(C2CCCC2)nn1)=O c1(C(N(C)CC2(CNC(C3(OC)CCC3)=O)CC2)=O)cc(S(N)(=O)=O)cnc1C N1(C(c2nnc(C(C)(C)C)s2)=O)CC2CCC(C1)N(C(=O)CCS(C)(=O)=O)C2 C(=O)(CCCCSC)NCC1(NC(C=CC(C)(C)SC)=O)CCOC1 Nc1c(C(=O)NCC(c2ccccc2F)NC(=O)Cc2ccco2)cccc1F c1(C(N2C(CNC(CCc3scc(C)c3)=O)CC(F)C2)=O)cc(C)nc(O)n1 CCCCC(CNC(=O)CSC1CCOC1=O)NC(=O)COC1CC1 CCCC(C)CC(=O)NN1CCCC1C(=O)NCC(Cl)Cl c1(C(=O)NC2(C(C)NC(C3CC(OCC)C3)=O)CC2)cncc(NC)c1 C(=O)(C1=NOC2(CCN(C(=O)CN)CC2)C1)N1C(C)C(=O)N(C)C1 C1(C(C)C)CCCC1C(=O)N(CCN(CCCN(C)C)C(=O)CC1CCC1)CCO C(C(=O)NC(C)CNC(=O)Cc1sc(C)nc1C)(C(C)(C)C)OC C#CCCCC(C)C(=O)NCCCCC(C)NC(=O)C(c1ccc(Cl)nc1)(F)F C1(NCc2[nH]nc(-c3cc(C)no3)n2)CCC(=O)N(CC(c2ccccc2)=O)C1 c1(OCC)cc(C(N2CC(C)(NC(C3CCN(CC(F)(F)F)C3)=O)C2)=O)sn1 c1(C(=O)Nc2cc(CC)cc(C(=O)COC)c2)nc2ncc(Br)cc2[nH]1 C(CCCC(=O)NCC(CO)NC(=O)Cc1cncnc1O)OCC C1(N(CCOC)C(c2csc(Cl)c2)=O)CCN(C(c2cnnn2C(C)C)=O)CC1 C1(CC)CC(C(N2CCC2C2CCCC2)=O)CCN1C(c1ccoc1)=O c1(N2CC(C(N3C(CN=[N+]=[N-])CC(F)C3)=O)C2)ccn2nccc2n1 C(=O)(CC(C(F)F)n1ccnc1)NCC(C)CN(C(=O)Cc1ocnc1CO)C C=CCCC(C(=O)Nn1cnnc1C)NC(=O)C1CCc2c[nH]nc21 Cc1cc(O)ncc1C(N1CCCC(C(C)NC(=O)CCc2ccncc2)C1)=O c1(C2C(SCCC(N3CC(CCNC(c4ccsn4)=O)C3)=O)C2)ccccn1 C1(NC(c2ccc(C(C)=O)o2)=O)CN(C(=O)C(O)CSC)CC1c1ccnn1C C1(CNC(CC2C(C)OCC2)=O)CN(C(=O)C(O)c2ccsc2)CC1(F)CO S(=O)(=O)(c1ccc(C(N2CC(NC(c3cc(OC)no3)=O)C(O)C2)=O)cn1)NC c1(C(N2CC3CN(CC(=O)Nc4nccs4)CC3C2)=O)ccc2nc[nH]c2n1 c1(OC)c(C(=O)NCC2C(C)CCN2C(c2cn(CC)cn2)=O)nc(O)nc1O CCC(CCCC(=O)NCCCC1CCOC1)NC(c1cc(C)nnc1O)=O C1(NC(C2ON=C(C)C2)=O)(CF)CCN(C(c2cc[nH]c2C2CCCC2)=O)C1 CC1OC2(C)CC1(C(=O)NCC(C)(C)NC(c1ccn(C(F)F)n1)=O)C2 c1(C(=O)NCCC2N(C(c3c(SC)snn3)=O)CCSC2)ccc([N+](=O)[O-])cc1 c1(NC(=O)NC(C(C)O)C)nc2c(s1)COCC2 N1(C(CC=CCC)=O)CCc2ccc(C(=O)NC3CCCN(C(C)=O)C3)nc2C1 C#CCC(C(N)=O)NCC1CCCOC1c1cnn(C)c1 c1(C(C)=O)cc(NC(C2OC3(C)CC2(C(=O)O)C3)=O)cc(C(C)C)c1.C1(C)CC1 c1(C(=O)NC(C2CN(c3ncnn4cccc34)C2)C)cnc2c(F)cccc2c1 Cc1cc(NC(c2cc(F)ccc2O)=O)ccc1NC(C1OCCN(C)C1=O)=O c1(C(C(=O)NCC=C)N(C2Cc3ccccc3C2)C)cnc2c(c1)COCC2 Cc1nn(C)c2c(N(C)Cc3ccncc3F)nc(=NCc3ccccn3)[nH]c12 c1(C(=O)NCC(O)CNC(c2sccc2C(F)F)=O)cc(O)nc2c1CCCC2 C1(OC)CN(C(=O)OC(C)(C)C)CCC1NC(C1CC(=O)N(C(C)C)C1)=O c1(C(=O)NCC2C(NC(C(=O)N(C)C)=O)C2)cc(CCO)on1 C1(NC(C(C2CCCCC2)NC(CC)C(N)=O)=O)CCCCC1c1ccccc1 C1(CC(=O)NCC(COC)C)CCN(Cc2cnn(C(C)C)c2)C1 C(=O)(C(F)CCCC)NC1(CC=C)CN(C(c2cncc(C(F)F)c2)=O)C1 C(=O)(C1=C(C)OCCC1)N1C(C)CC(NC(C=CCC)=O)C1 C1(n2cc(CCC(C)O)nn2)CC2CCC1(NC(=O)Cc1cnc(O)nc1O)C2 c1(C(=O)NCC(CC)(C)NC(=O)CC2CCCOC2)nc(Br)sc1C C(=O)(C1=C(Cl)CCOC1)N1C(C(=O)NC2(C(N(C)C)=O)CC2)CC(F)CC1 C1(COC(C2CCCN(C(C)C)C2)=O)CN=C(c2ccccc2)N1 C1(NC(C2OCCN(CC)C2)=O)CC12CCN(C(=O)CN1CCCS1(=O)=O)CC2 c1(SC)ccc(N2CCN(C(C3CCC(C(N)=O)O3)=O)CC2)cc1 CC1=NOC(CC(=O)NC2(C(=O)NC3(c4ccccn4)CC3)CC2C)C1 C1(CNC(C(C)O)=O)C2CC1N(C(c1cccc(NC(=O)NCC3CC3)c1)=O)C2 c1(CNC(CCCNC(N)=O)=O)cccc(CNC(=O)C(F)CC2CCOC2)c1 C=CCC(F)(F)C(=O)NC1CCC1NC(=O)CC1CCN(OC)CC1 c1(NC(=O)C(N2CC(O)(CC(N3CCCC3)=O)C2)=O)ccc(C(=O)CF)cc1 C1(Cc2cn(C(C(=O)OC)C)nn2)CCCCN1C(c1ccnnc1)=O c1(CC)ncoc1C(=O)NC1CC(NC(=O)CCCOC(C)=O)C1 CC1CN(C(C2(O)CCC2)=O)CC1C(N1CC(N2CCC2)C1)=O N1(CCCNC(=O)NCc2cc(OCC)n[nH]2)CCOC(C)C1 c1(C(=O)NCCC(C)(C)NC(=O)C(O)C(C)(C)C)nccn2c(Br)cnc12 c1(C(=O)OCC)ccc(C(=O)Nc2cnnc(I)c2)cc1 C1(NC(=O)CC2CC2(Cl)Cl)CC2(C1)CC(NC(C1CC(N3CCCC3)C1)=O)C2 C1(CNC(C2C(C(=O)OC)C2)=O)N(C(C2CCC3(CC2)CC3)=O)CCCC1(C)C Cc1cc(C(C)NCCCOCCNC(=O)OC(C)(C)C)cc(C)c1 CC(F)CC(=O)NC1(CNC(=O)C(C)CSCc2ccccc2)CCCC1 c1(C(C)Nc2ccc(C)cc2O)ccc2c(c1)OCCCO2 CCC(C(=O)N(CCC(C)(C)NC(=O)Cc1sccc1C)C)NC(C)=O N#Cc1ccc(F)c(C(N2CC(C3(NC(C4C(C5CC5)C4(F)F)=O)CC3)C2)=O)c1F c1(OC)cc[n+]([O-])c(C(=O)NC2CN(C(C3CC(F)C3)=O)C2)c1 Cn1cc(-c2cc(C(N3CCC(NC(=O)C(c4cccnc4)O)C3)=O)on2)cn1 N1(C(c2cc(COC)on2)=O)CCC2(CC1)CC2(C)C(=O)NCC1CC1 N1(C(C(CC)C)=O)CC(OC)C(NC(C2(c3ccccc3Cl)CC2)=O)C1 C1(C(=O)NCC2N(C(C(C)C3CCCO3)=O)CC2)(CF)CC2(CCC2)C1 c1(NCCn2c(C)cc(C)n2)ncccc1S(=O)(=O)N1CCC2CC12 c1(C(=O)NC(CN(C(C(CC)C(C)C)=O)CC)C)ccc([N+](=O)[O-])cc1C N1(C(c2cc(C)[nH]n2)=O)CC(NC(c2ccc(C)o2)=O)C2CC2C1 n1(C(CC)C)nc(CCC(C)C)nc1-c1csc(C)n1 c1(C(C(=O)NC(c2nc(COCC)on2)C)OCC)ccc(Cl)c(Cl)c1 N1(C(CCCC=C)=O)CC2(CCN(C(=O)C(O)C(C)CC)CC2)C2COCC12 C=CCCCC(C(=O)NCCCCCCF)NC(C1CCO1)=O c1(C(N(C2CCN(C(=O)CCC3CCCCCC3)C2)C)=O)ccn2ncccc12 Cc1nc2[nH]c(C(=O)NC(C)CN(C)C(c3ccc(C4CC4)nn3)=O)cc2s1 C(N=c1[nH]cncc1F)C1(NC(c2cnc(-c3ccccc3)nc2)=O)COC1 N#Cc1ncn(CCCC(=O)NCCCNC(=O)CCc2cn[nH]c2)n1 N1(C(C(C(=C)C)(C)C)=O)CC2(C1)SCCC2NC(C1CC1OC)=O Cc1nc(N2CCN(CC3CCNC3)CC2)nc2c1CCCC2 N1(C(C(CC)n2cccn2)=O)CCN(C(=O)COc2cccnc2)CC1CCC CCCC(O)CC(=O)NCC1CCC(NC(c2nnn3c2CCC3)=O)CC1 N1(C(C2(C(C)C)COC2)=O)CCCC(C)(C(N2CCC(F)(F)C2)=O)C1 Cc1ccc(C(=O)NCCC(O)CNC(=O)Cc2ccnn2C2CCOCC2)s1 Cc1ccc(C(N2CC3CC2(CNC(C2CCN2C(C)(C)C)=O)C3)=O)c(N)c1 C1(C(N2CC3C(NC(C(C)OCC#C)=O)C(C3)C2)=O)C2CCCCCCC12 c1(OC)c(C(=O)NC2CN(C(c3cc(Br)co3)=O)CC2C)cc(F)cc1F C1(CCNC(C2(C=C)CCC2)=O)CN(C(=O)Cc2[nH]cnc2C)CCCO1 C1(C(=O)OC)(NC(=O)CSCC2CCS(=O)(=O)C2)CC2(CC(C(F)(F)F)C2)C1 N1(C(C)=O)CC(C)(C)OCC1CNC(=O)Nc1cc(C#C)ncc1 c1(C(=O)NC(C2CCN(C(=O)CC3(C)CCOCC3)C2)C)cc2c([nH]1)CCCC2 N1(C(CCCSC)=O)CCC(Nc2nc(C)cc(C)n2)CC(C)(C)C1 C1(CC)CC(C(=O)N(CCNC(=O)C(=O)NCC(F)(F)F)CC2CC2)CCO1 c1(C(C)C)ncc(C(N2CC(OCCNC(=O)C(C)(C)c3ccns3)C2)=O)[nH]1 Cc1ncc(C(=O)NCCOCCCN(C(=O)CC(F)(F)F)C)cn1 N1(C(C(CC#C)O)=O)CCOC(C)C1C(=O)NC(c1ccsc1)C C1(C)(CNC(COc2cn(C(C)S)nc2)=O)CCCN1C(c1csc(=NC)[nH]1)=O c1(C(=O)NC2C(NC(Cc3cc(C)sc3)=O)C2)cc(Br)c(C)cc1F C#Cc1ccc(C(=O)NCC(C)N(C)C(C2CCc3ncsc3C2)=O)cc1C C1(CC(N2C(C)C(NC(=O)CCC3CCC3)CC2)=O)OCCCC1(C)C C(C)(C)(CCCNC(=O)COc1cccc(F)n1)NC(C(CC)=CC)=O CCC(CC)(CCNC(=O)C(C)Cc1c(C)n[nH]c1C)NC(c1ccsc1C)=O CN1CC2(CN(C(c3cnc(CNC(c4ccnn4C)=O)nc3)=O)C2)C1 C1(NC(c2c(-n3cc(CNC=O)nn3)cccc2)=O)CC2CCCC2C1 C1(C(N(C(CCNC(COCCC=C)=O)C)C)=O)CCN(C2COC2)C1 c1(CC2N(C)CCC2)nc(-c2ccc(C3CC3)cn2)n(C2CCC(C)(C)C2)n1 c1(N2CCC(C(=O)OC(C#C)CC)C2)ccccc1Cl CCC(O)C(C)(C)C(=O)N1CCC(CCOC)(NC(=O)CC2CC=CC2)CC1 c1(N2CCN(C(CCNC(C3C(C)C3)=O)=O)CC2)ccncc1C#N CCCC(CCC)C(=O)N1CCC(CO)(NC(C2CC3C(C2)C3(F)F)=O)C1 Cn1c(C(=O)NCCC2(O)CCCN(C(C3(C)CSC3)=O)C2)cc2occc12 N1(C(c2cc(C(C)C)nn2C)=O)CCC(C)CC1CNC(=O)CC1CC12CC2 c1(C(=O)NC2C(CNC(C3CCC(C(C)C)CC3)=O)C2)cc(Cl)c(F)c(Cl)c1 c1(C(N2CCN(C(C3C(COCC)C3)=O)CC(CO)C2)=O)cccc(C)c1[N+](=O)[O-] c1(C(N2CC3C(NC(c4cccc(Cl)c4F)=O)(C3)C2)=O)cccc2[nH]ccc12 N1(C(C2(C)CCC2)=O)CCC2(CC1)CC2NC(C1CS(=O)(=O)C1)=O c1(NC(C(C=CC)O)=O)ccc(Cl)c(C(=O)NCC2CC2)c1 C1(NC(COCC(=C)C)=O)COC2C(NC(c3nnsc3SC)=O)COC12 C(=O)(C1=CS(=O)(=O)CCC1)NC(C(C(C)C)NC(=O)Cc1csc(C(C)C)n1)C C(C1(C)CCOCC1)=CC(=O)NCc1cccc(C(NOCC(C)C)=O)n1 C#CCC(CC(F)F)NC(c1n[nH]cc1CNC(=O)C(O)C1CC1)=O c1(C(=O)NC2CC(NC(C(C)OCC(F)(F)F)=O)CC2O)nc2c([nH]1)CCCC2 C(=O)(CS(=O)(=O)C(C)(C)C)N1CCC(C)(CNC(C(C)N(C)C)=O)CC1 C(CC(CO)C(C)C)NC(C(C1CCC1)NC(c1c(CC)ncnc1)=O)=O c1(C(=O)OCC2(C)CC(C)C2)cnn(-c2ccc(Cl)cc2)c1C(F)(F)F O=C1CCC2(CCN(C(C3CCCN(c4cc(C(=O)O)ccn4)C3)=O)C2)N1 c1(CNC(C2CCC(C(C)NC(C)=O)C2)=O)cc(OC(F)F)n(C)n1 C1(CNC(c2c(CC)ocn2)=O)CCN(C(c2cc(C3(C)CC3)on2)=O)CC1C C1(NC(c2c(OC)nc(C)cc2)=O)CCSC12CN(C(=O)CN(C1CC1)CC)C2 C(=O)(CCCCCCCS(C)(=O)=O)NC(CC)CNC(C1CCN(OC)CC1)=O N1(CC(N2CCC(OCCNC(CC3(COC)CC3)=O)C2)=O)CCC(C)(C)C1 C1(C(N2CC(CNC(CCc3cccc(C)c3)=O)C2)=O)CCCC(C#N)C1 Oc1ncc(CN(C2COC2)Cc2ccco2)s1 c1(C(=O)NC2CCC(NC(C3(CC4CC4)CCC3)=O)C2)cc2c(o1)CCCC2 CC(CCC(F)(F)F)NC(C1(CCNC(C2CC(F)C2)=O)CC1)=O N1(C(C(CCN(C)C)NC(Cc2c(C)n(C)cn2)=O)=O)CC2CC3CC2C1C3 C1(O)(CN(C(C2CS(=O)(=O)C2)=O)Cc2ccncc2)CCNC1 O(NC(=O)CCN(C(=O)Cc1ccsn1)CCO)CC(C)O C1(C(NOCCC=C)=O)CCN(C(=O)CC(O)C(C)C)CCO1 C1(C(N2CC3C(NC(c4ccc(COC)[nH]4)=O)(C3)C2)=O)CCc2[nH]nc(O)c2C1 C1(C(N2CCC(CCC(=O)N(C)CC3CC(=C)C3)C2)=O)(COC)CCCC1O C1(CNC(C(=O)NCCCCC(N)=O)=O)OCC2CCC1C2 C=C1CCC1C(=O)NCCC(C)NC(=O)C(C)N(C)C C(=O)(C(O)CC[S+](C)C)N(C)CCNC(=O)C(c1ccccc1Cl)(C)C c1(NC(C2N(C(c3cc(OC)n(C)n3)=O)CCOC2)=O)cc(F)ccc1[N+](=O)[O-] Cc1ncc2ccc(C(N3CCCC(O)(CNC(=O)CCC4(C)CC4)C3)=O)cn12 c1(CNC(=O)CCOC2CCC2)cn(C2CCN(C(c3ccc(Cl)o3)=O)C2)nn1 CC(C)CC(C)(O)C(=O)NC1CC=CCC1C(N1CC(F)CC1C)=O C1(C2CCCO2)(C(=O)NCC(CC)NC(=O)C(C)c2ccsn2)CCCC1 C1(C(=O)NC(C2(O)CCN(C(c3c(C)occ3)=O)CC2)C)CCCCC(F)(F)C1 c1(C(=O)NC23CCC(C2)N(C(c2cncnc2)=O)C3)cc(Cl)cc2ccccc12 C12(NC(c3ccc(C)cn3)=O)CCCC1CN(C(C13COC(CF)(C1)C3)=O)C2 C(C1=NOC2CN(C(c3nn[nH]c3Cl)=O)CC12)NC(c1cc2nc[nH]c2cn1)=O Cc1nc(C)c(CNC(=O)C(=O)NC(C2(C)CC(F)(F)C2)C)s1 c1(-c2ccc(S(C)(=O)=O)nc2)ccc2nc(O)cc(C(=O)NCC(N)=O)c2c1 c1(CCOC)cc(C(=O)NCC=CCNC(=O)CCc2ccc(C)s2)no1 C1(C(N(CCCC)C(C)CC)=O)CN(C(=O)C(F)C(C)(F)F)CC12CCC2 C(c1ccc(F)cc1)=CC(=O)NC(CNC(CC(C)SC)=O)(C)C C1(NC(=O)Cn2ncc(SC)n2)CN(C(=O)C(C)NC(=O)OC(C)(C)C)CC1F Cc1nn(CC(=O)N(C)CC2CCCN(C(=O)C3=CCSC3)C2)c(C)c1C=NO c1(C(N2CCC(C)(CNC(CCCCC)=O)C2)=O)cc(Br)cc(Cl)c1C CC1(C)CCN(C(=O)Cc2ccon2)CC1CNC(C1(C(N)=O)CC1)=O C(C(C)(O)CC(=O)N1CCC(CNC(c2cncnc2)=O)C1(C)C)OC C1(O)(CNC(C=C2CCN(C)CC2)=O)CCN(C(C2CS(=O)(=O)CCO2)=O)CC1 N1(C(CCCN(C)C)=O)CC2(C=C(C(=O)N3CC(O)(CCO)C3)CO2)C1 C(=O)(CCCCC(=O)N=C1CCN(C)N1)Nc1ccc(C(C)(C)C)cc1 C(N=c1[nH]c(=NCc2nc(CO)cs2)[nH]c2c1CCCC2)c1c(C)ccc(C)c1 c1(C(N2CC3C(NC(C(C)C(F)F)=O)C3C2)=O)cnc2c(c1)CCS(=O)(=O)C2 c1(C(=O)NC2C(NC(c3cncc(F)c3)=O)CCCC2)oc2ccccc2c1Cl C(C(C)(C)C(=O)N1CCCC1CN(C)C(c1cccn1C)=O)N(C)C C1(C(=O)NC2(C)CN(C(C(C)CSc3ccccc3)=O)C2)CCOC(=O)CC1 N1(C(c2c(C)ncn2O)=O)CCCC2(CCC(NC(c3cnn(C)n3)=O)C2)C1 C1(C(=O)NCCCCNC(C23CC(C)C2C3)=O)CCN(C2COC2)CC1 c1(NC(C2CC(C(=O)OC)C2)=O)ccc(S(=O)(=O)Nc2ccccc2Br)cc1 N1(C(C(C#C)(C)C)=O)CC(CC(N2CC3CC2CS3=O)=O)C2(CC2)C1 n1(CC)cc(CC2(CCNC(=O)C=CCOC)CC2)nn1.C1(C(=O)NC)(OC)CCC1 N1(C(C(CC#C)C)=O)CCN(C(c2cn(C)nc2Br)=O)C(COC)C1 CC(C)CC(F)C(=O)NC1C2CN(C(=O)C3=COCCC3)CC12 N1(c2nnc(C)c(C)n2)CCCC12CCN(C(C1CCC(C)(C)C1)=O)C2 CC(C)(C)C(C)(C)C(=O)NCCOC1CCN(C(C2CC(F)(CO)C2)=O)C1 c1(C(N(CCNC(Cc2c(C)n(C)cn2)=O)CC2CC2)=O)cnc(O)c(F)c1 N1(C(c2n(C)ccc2)=O)CC(NC(c2ccc(Cl)nc2)=O)C(C#N)C1 C1(CCNC(C(C)(C)OC(C)C)=O)CN(C(c2cnn(C3CC3)c2)=O)CCO1 CS(=O)(=O)CC(=O)N1CC(O)(CNC(=O)C(F)n2ccnc2)C1 CCC(CC)(CC)C(=O)NCCCCC(=O)N(C)Cc1sccc1C N1(C(C(C(=C)C)(C)C)=O)CCC2CN(C(c3ccoc3Cl)=O)C2C1 CC(CC(=O)NC1(C2CN(C(=O)CC3(C)CCOCC3)C2)CC1)C(C)(C)C N1(C(c2cn(C(C)C)nn2)=O)CCN(C(=O)C(O)C(F)(F)F)CC(O)C1 O=C1COC(CNC(C2CC(O)CN2C(=O)CCc2ccccn2)=O)CN1 CC1(C(=O)NCc2c[nH]nc2C(=O)NCC(O)C(N)=O)SCCCS1 c1(OC)ccc(OC)c(C2=NOC(C(=O)Nc3ccc(F)c(SC)c3)C2)c1 Cc1cc(C#N)nc(=NCCC2CCCN(C(c3c(F)ccc(F)c3F)=O)C2)[nH]1 C(=O)(CC(C)(C)C#N)NCC1(F)CC(CNC(CCn2c(C)nc(C)n2)=O)C1 C(C)(CO)(CN=c1[nH]c(=NCC2CCCCN2C)c2cc(F)cc(F)c2[nH]1)OC N1(C(c2cc(C(F)F)cs2)=O)CCCCC1Cn1cccn1 c1(C(N(c2nc(C)cc(OC)n2)CC2(OC)CNC2)=O)ccc([N+](=O)[O-])c(C)c1 c1(C(=O)NCC2CN(C(CC3(C)OCCO3)=O)CC2O)ccc2nnc(O)n2c1 N1(C(C(CC=CC)C)=O)CCOC(C(N2CC3(CCC3O)C2)=O)CC1 c1(C(=O)NC(C)CCNC(C2C3COCC23)=O)ccc(-c2nncn2C)cc1 N1(C(CC(CC)C2CC2)=O)C2CCC1CC(CCNC(c1cccn1C)=O)C2 C(CCCCC(=O)NCC1CCC(C)N(C(C2CC(O)CN2C)=O)C1)OC c1(CC(=O)NC2CC(CNC(CCCC(=O)NCC)=O)C2)ccc2c(c1)OCO2 c1(C(=O)NCC2(O)CC(NC(C(C=C)(C)O)=O)C2)cc(C)n(CC(F)(F)F)c1C CC1(NC(c2cccc(F)c2N)=O)CCCN(C(C2CCC3(CCC3)O2)=O)C1 N1(C(C(CCC)OC)=O)CCN(C(c2[nH]ccc2-c2ccccc2)=O)CC1C N1(C(C2(C=C)CCN(C(=O)C=CCN(C)CC)C2)=O)CC2CC(C1)N(C)C2 C(=O)(CC(O)CCC)N1CC(CC=C)(NC(=O)C(n2nc(C)cc2C)C)C1 C1(C(=O)NCC2CC(F)(CNC(CS(CC)=O)=O)C2)CC(F)(F)C1(C)C C=CCCCCC(=O)NCC(CNC(c1cc(OCC)ccc1N)=O)OC c1(C(=O)NC2(CCNC(CCc3c(C)noc3Cl)=O)CC2)cc2c(s1)CCSC2 N1(C(C(C)n2ccnn2)=O)CCN(C(c2ccccc2CO)=O)CC1CC(F)F C(CC(C)(C)C(=O)NCC(C1CCC1)NC(=O)C(C)(C)c1ccccn1)SC S(=O)(=O)(c1c[nH]c(C(N2CCCC(NC(=O)C(C)(C)C)C2C)=O)c1)NCCOC c1(C(c2n(CCOC)nnn2)NC2CSCCSC2)cccc2c1CCC2 C(=O)(C(C)CC(C)(C)C)NC1C2CN(c3c(CC)c(Cl)ncn3)CC21 c1(SC)cccc(C(=O)NC(C2CC2CC2(NC(=O)NSC)CC2)=O)c1.C1CC1 C=CC1CCCN(C(=O)CC2CCN(C(=O)C(C)(C)CCC)C2)C1 c1(C(=O)NCC2CN(C(CCCN(C)C)=O)CC2(C)C)ccc2nc[nH]c2c1F N1(C(c2nc3cnccc3s2)=O)CCC2C(CCN2C(c2cccc(O)n2)=O)C1 C1(NC(c2n(Cc3nnn(C)n3)nnn2)(C)CC2CCCC2)CCC(=O)NC1 Cc1nnc2n1CC(C(=O)NCC=CCNC(C1(CF)CC1(F)F)=O)CC2 c1(C(=O)NCCC2(NC(CC=CC=C)=O)CC2)nc(C)oc1C C1(NC(=O)CCC2CCN(C(=O)COC34CCC(CC3)C4)C2)CCOC(=O)CC1 c1(C(N2C(CNC(CS(CC)=O)=O)CC2)=O)c(SC2CCCC2)cccc1F C1(N(C(C2ON=C(CC)C2)=O)C)CCCN(C(C2(C)CCC(=O)N2)=O)CC1 C1(C(C)NC(c2sccc2C(N)=O)=O)CCCN(C(C2(CF)CCC2)=O)C1 C1(C)(NC(C(c2ccccc2Cl)C)=O)CCN(C(c2scnc2Cl)=O)C1 C(=O)(C1CSc2ccccc21)NCCCN(c1cc(C2CC2)ncn1)C(C)C C1(CNC(=O)C(F)F)CN(C(c2sccc2SC(F)F)=O)CC12CC2 c1(C(=O)OCC)cnc(Cl)[nH]c1=NCCOCCC1CCCO1 CCC(N=c1nc2c(cnn2C)c(NCC2CC(=O)N(C)C2)[nH]1)C1CCCC1 Cc1oc(Cl)nc1C(=O)NC1(CNC(C2CCCNC2=O)=O)CCOC1 N1(C(CNC(c2cnc(I)cn2)=O)=O)CC(C(=O)Nc2ncccn2)CC(F)C1 C(=O)(C(CNC(=O)CCCn1cccn1)C(C)(C)C)NC(C#C)(C)CC c1(C(=O)NC2CN(C(COc3cc(C)on3)=O)CC(F)C2)ccc2scnc2c1 NC(=O)C1=NOC(CNC(=O)CC2CC(NC(C3(CF)CC3)=O)C2)C1 c1(C(=O)NC(CNC(C(CCCOC)C)=O)(C)CO)cccc2nccn12 CC1(C)CCCCCC1NC(C1(C)CC(O)CN1C(C1CC2(CC2)CO1)=O)=O CC1CN(C(c2n[nH]cc2Cl)=O)CC(C)CN1C(c1ccc(F)c(C2CC2)c1)=O c1(C(N)=O)ccc(C(=O)NC2CN(C(c3cccs3)=O)C2)cc1 N1(C(C=CC=CCC)=O)CC2CCCC1C2CNC(=O)C(n1cc(C)cn1)C C(=O)(C(O)CCNC(=O)N(C1(c2ccncc2F)CCC1)C1CC1)OC Cc1ccc(Cn2nc(-c3occc3C)nc2-c2ccc(CC3CCC3)o2)cc1 c1(CC(=O)NC2CCN(C(CCC#C)=O)CC2F)nn(C)c2ccccc12 N1(C(C(C)C(C)(F)F)=O)CC(NC(c2ccc(F)c(F)c2)=O)Cc2ccccc21 N(C(=NCCC1CCS(=O)(=O)C1)NC1CCCC(C)(C)C1)CCC(=O)NC N(C1COc2ccccc21)C(C(=O)NC(C=C)C1CC1)=O CCC(C(=O)NC12CN(C1)C2)n1nccc1C.C(C)(C(C)C)=CC(=O)OC CCCCCN(C(=O)CC1(NC(=O)CSc2nc[nH]n2)CCC1)C c1(OCC)cc(N2CCCCC2CNC(=O)C=C(Cl)Cl)ncn1 c1(C(=O)NCCC(CNC(C(C)SC(C)C)=O)O)cccc2oncc12 C(=O)(C(C)CC(C)(C)C)NC1C=CCC(C(=O)NC2C(C)NC(=O)CC2)C1 C1(NC(c2ccc(SC(C)C)cc2)=O)CCC12CN(C(c1nocc1Cl)=O)C2 CC1(O)CCCN(C(C2C=CCN(C(C3C4(CC4)C34CC4)=O)C2)=O)C1 C1(NC(C(CN(CC)CC)F)=O)CC12CC(NC(=O)CNC(c1ccoc1)=O)C2 Cc1cc(Cl)c(C(=O)NC2CCCC(CNC(c3ccn(C)n3)=O)C2)cc1C c1(C2(C(=O)NCCC(C)NC(=O)CC34CCCC3C4)CC2)ccccc1F CCCC(F)C(=O)NC1CN(C(=O)CC2CC(C)C2)CC1CCC C1(O)(C(CNC(CCCNC(C)=O)=O)C)CCN(C(=O)CN2CCCC2=O)C1 C1(C(N(C(C=C)C2CC2)C)=O)CCC(C)N(C(=O)CCCSCCC)C1 c1(C(N(C2CCCN(C(=O)CC3CCCSC3)CC2)C)=O)cccc(F)c1Cl C(=O)(CC(C)(C)COC)N1C(CC)C(NC(=O)C(c2cccc(OC)c2)O)CC1 N1(C(C=C2CCN(C)C2)=O)CCC(NC(=O)C(c2cc(F)cc(F)c2)O)C(F)C1 CC(C)(C)[Si](C)(C)Oc1cccc(NC(=O)NCC2CC2C#N)c1 C1(C(N(CCC(=O)N)C)=O)CCCC12CCC2.C(CCC(=O)NCC1CC1)NC=O c1(C(=O)NCC(C)(C2CCC2)NC(C(CCC)N(C)C)=O)n[nH]c2cccnc12 c1(C(N2CCC(C(C(=O)NCCC(C=C)C)C)C2)=O)cc(C)n(C)c1C CCC(C)(O)C(=O)NC1CCN(C(=O)Nc2ccco2)CC1.C1(=O)COCCN1 C=Cc1ccc(C(=O)NCC(C)(CC)C(=O)N2CCC(C#N)CC2)cc1 C(CN=c1cccc(S(=O)(=O)NC2(C)CN3CCC2CC3)[nH]1)NS(CC)(=O)=O C1(CNC(=O)CC2CCOC2)C=CCN1C(c1ccc(-c2cccs2)s1)=O C(C(=O)N1CCCO1)NC(CC(CC1CC1)NC(C1(C)CC2CC2C1)=O)=O C(=O)(C1=NN(C)C(=O)CC1)NCC(C1CCC1)NC(c1c(OC)nsc1)=O CC(CNC(C1CC=CC(O)C1)=O)CC(=O)NCCCCO c1(C(=O)NCC2CCC(C(=O)NCC3CC(=O)NC3)CC2)cc[nH]c2nccc1-2 C1(CNC(c2c(C)ccnn2)=O)CC(NC(=O)C#CC(C)(C)O)C12CCC2 C(C)(C(O)C(=O)N1CC(N2CCN(C(c3cscn3)=O)CC2)C1)SC C1(C)(CNC(C=C(C)C(F)F)=O)CC(NC(c2cc(-c3ccncc3)on2)=O)C1 N1(C(C=CCN(C)CC)=O)CCC2(CC1)CC2NC(c1ccc(N(C)C)cc1)=O CC(C)(CNC(=O)CC1COC(=O)C1)CC(=O)NC(c1ccccn1)CO c1(C(=O)NCC(C)(CO)NC(c2ccc(C(C)=O)[nH]2)=O)cc2cccnc2o1 N1(C(C(CC#C)C)=O)CCC2C(CCN2C(=O)C(c2c(C)cccc2C)=O)C1 CC(C)CC(C)C(=O)N1CC(=O)CC1C(=O)NCCN1CCCOC1=O CC(c1cccnc1)=CC(=O)NC1CCCC1NC(=O)CCNC(=O)C=CCl C1(CC)C(NC(c2cncc(F)c2)=O)CCCN1C(c1ncn(C)c1C)=O C1(C(=O)OC)CCC(CC(=O)NC2(CCNC(c3csc(Cl)c3)=O)CC2)CC1 C(=O)(C(O)C(F)(F)F)N(CCC(C)NC(c1cc(CN(C)C)on1)=O)C C1(CC(=O)NC(CC(=O)NC(c2nc(=O)o[nH]2)C)C2CC2)CCN(C)C1=O C1(CN(C(CCCSCC)=O)CC)CCN(C(=O)Nc2ccsn2)CC1 C(=O)(C(O)CC(C)C)N1CC2C(CNC(C3(CCOCC)CCC3)=O)(C2)C1 CC1CCCC(CC(=O)NCc2cn(Cc3nc(C(=O)O)cs3)nn2)C1 c1(CCC(=O)NC2C=CCN(C(C3C(C)(C)OCC3)=O)C2)cc2ccccc2o1 Cc1cccc(C(CO)NC(C2CCCCN2Cc2nc(Br)cn2C)=O)c1 N1(C(=O)CC2CC2)CCC2CCN(C(C3(CCF)CC3)=O)CC2C1 N1(C(c2nc(C)oc2)=O)CCC(NC(c2cc3c(ncn3C)s2)=O)C2(CCC2)C1 c1(C(N2CC3CCN(c4ncncc4F)CC3C2)=O)cc(Cl)c(Cl)c(Cl)c1Cl C1(CC(=O)N(C2CCN(C(c3nc(=O)n(C)[nH]3)=O)C2)CCC)C=NN(C)C1=O C(=O)(C1=C(Cl)CCOC1)N1CCN(C(c2c(C)nn(CCO)c2)=O)C2C1C2 Cc1cccc2c1CN(C(=O)C(F)CC1CN(C(=O)CC3OCCC3(C)C)C1)C2 c1(C(=O)NCC2(NC(CC=C)=O)CCCCC2C)cnc2n(c1=O)CCS2 C1(C(=O)NCCC(CC)(C)NC(=O)CC2CC2)Cc2cscc2C1 c1(OC)cccc(C(=O)NC(C)CC2CN(C(=O)CC#N)C2)c1OC C(=O)(CC(C)C(F)(F)F)N(C1CCN(C(=O)CSC(C)C)CC1)CCOC C=CCC(CC(C)C)C(=O)N(C1CN(C2CC2Nc2ncoc2C(F)(F)F)C1)C c1(C(N2CC(N(C(c3c(C)noc3)=O)C)C(O)CC2)=O)cnn2cccc2c1 N1(C(C(C)OC)=O)CC2CCC1CN(C(=O)COCC(F)F)C2 c1(C(C)CC(=O)Nc2cnn(-c3ccccc3F)c2)ccc2c(c1)OCO2 C1(NC(c2ncn(CC)n2)=O)C=CCN(C(c2cnc(O)o2)=O)C1 CC(CNC(=O)C(C1(O)CCCC1)F)C(=O)N(C)CCN(C)C1CC1 O=C1CCC2(CN1)CN(C(=O)CSCCNC(C1CC3(CCC3)CO1)=O)C2 C1(C#N)(C(N2CCC(CN(C(=O)COc3ccn(C)n3)C)C2)=O)CCCC(=O)C1 C1(CC(=O)NCCOC2CCN(C(c3cnc(CCC)s3)=O)C2)CC2(CCC2)C1 C1(OC)CC(CCNC(C2C(C)(C)C2(F)F)=O)N(C(=O)C=Cc2scnc2C)C1 c1(C(=O)NCCC2CN(C(=O)COC(F)(F)C(F)(F)F)C2)n[nH]c2c1NCCC2 N1(C(C(CCC)C)=O)CC(C(=O)Nc2cc(CO)ccc2O)CC(F)C1 CC1C2C(CCN2C(=O)CC2CCCCC2)CN1C(=O)C(=O)N=S(C)(C)=O N1(C(C(C)CC2CCCCC2)=O)CCC2(COC(CNC(=O)CC3CC3)C2)C1 c1(OC)cc(NCc2cc(-c3cc(C)n(CC)c3C)no2)cc(Br)c1.[SH](C)(=O)=O C=C(C)C1OCCC1C(N1CCC(CO)(NC(=O)CN2CCCCCC2)CC1)=O C1(CC)CN(C(=O)CS(=O)(=O)N2CCCCC2)CC1NC(c1cnn(C)c1)=O N1(C(C2(C(=O)N(C)C)C(C)C2)=O)CCN(C(=O)CCc2cn(C)nn2)C2COCC12 C1(NC(C)=O)CCC(O)CN(c2cnc(Br)c(Br)n2)C1 c1(C(C)Nc2nc(COC)nc(N3CCCC(O)CC3)c2)cccc2c1OCO2 C1(C(=O)Nc2cc(C)cc(C)c2)N(C(C2CCC3(CCC3)C2)=O)CC12CCCC2 C1(C(=O)NCC(CNC(CSCC)=O)F)COCC1n1ccnc1 C(CNC(C1(Cl)C2CCC(=O)C12)=O)(CC(F)(F)F)NC(c1csc(O)n1)=O C1(C(=O)NC2CC(CCNC(C(CCCC)O)=O)C2)CCc2nnc(C)n2C1 c1(C(N2CCC(C)(NC(=O)CCSC(F)(F)F)C2)=O)ccc2cccnc2n1 Cc1cc(OCC(=O)NC2CCC3(CC2)CC3)ccc1F Cc1nc2c(C(=O)NCCC(C(C)C)NC(=O)C=CI)ccnc2[nH]1 c1(C(=O)NCC(c2ccc(F)cc2)NC(CCOCCC)=O)nc(Cl)c(CC)[nH]1 C(=O)(CC(C)(C)C(C)(F)F)N(CC(CNC(Cc1ccc(OC)cc1C)=O)C)C c1(OCC=C)cccnc1CN1CCC(c2ccccc2)(CO)C1 CC1CN(C(C2CN(C(=O)CCCC#N)CC2(F)F)=O)CC(C)(C)CO1 c1(C(C(=O)NCCCC)N(C(CC)C2CC2)C)cccc(CC2CC2)c1 C1(CC=C)(C(=O)N(C)CC2CCCCC2)CCCN1C(=O)CC(=O)NC1CC1 c1(C(=O)NC2CN(C(CC=CC)=O)CC2CC2CC2)cnc(CO)nc1C N1(C(=O)NCc2cccc(OC(C)C)c2)CCc2ccc(CC)cc2C1 CC1CCC(NC(c2[nH]nnc2C2CC2)=O)CN1C(C1CCCC(C)(C)C1)=O c1(NC(Cc2nc(-c3cccc(C)c3)sc2)=O)ccc2c(c1)OCCN2C c1(OC)ccnc(OC)c1C(N1CC2C(CNC(C3CCC(C)(C)C3)=O)C2C1)=O C1(C(=O)NC(CC)Cc2cccc(Cl)c2)CCN(C(=O)OC(C)(C)C)C1(C)C c1(C(c2ccc(F)cc2)NC(=O)NC2(C)CSC2)c(F)cccc1F c1(NCc2ccc(C)cc2F)nc(N2CCN(C3CCC3)CC2)nc2scnc12 c1(C2(C(=O)NCCN(CCC)C(C3CCC(=O)O3)=O)CCC2)ccc(F)cc1F O=C1COc2cc(C(=O)NCc3cccn4c(Br)cnc34)cnc2N1 CCC(CCOC)C(=O)N1CCN(C(=O)C=CCOC(C)(C)C)C(C2CC2)C1 N1(C(c2cc(C(N)=O)ncc2)=O)CC2(CNC(C3(C(F)F)CC3)=O)CCC1CC2 N1(C(Cn2ccc(C)n2)=O)CC(CC(=O)NCC(C)S(N)(=O)=O)CC1(C)C c1(C(N(CC)Cc2cc(C)c(Cl)s2)=O)cc2c(nn1)OCCS2 N1(C(C2N(C(C(CCC)NC(N)=O)=O)CC(C)C2)=O)CC(O)CC(O)C1 C(=O)(CS(=O)(=O)C(C)(C)C)NCC(CNC(c1c(CC)cccn1)=O)(C)C N1(C(=O)CCc2ccc(F)nc2)CC2(CCCCN2C(=O)CC2CCC3CC23)C1 c1(NCCOC2CN(C(=O)NC)C2)n[nH]c2c1CC1CC21.C12(CC1)C(=O)N2 Cc1cc(CCC(=O)NC(C2CCCC2)CNC(=O)C(C)CSC(F)(F)F)n[nH]1 C1(CC(=O)NCC2C(OC(C)=O)CCC2)C2CCC(C2)N1C(=O)CC1(C)CC1 C1(CCCC)CN(C(c2cnn(CC)c2)=O)CCN1C(=O)C(C)CC(=O)OCC C(CNC(=O)C(C)C#N)(CCNC(=O)CCc1ccoc1)OC Cn1ncc2c(N3CC(CO)OC4(CCC4)C3)nc(=NCc3cnc(O)[nH]3)[nH]c12 c1(CCNC(C2C3N(C(=O)OC(C)(C)C)C(CC3)C2)=O)c[nH]c2cccc(Br)c12 C1(C(N(C(CF)C(F)(F)F)C)=O)CC(C)(C)CCN1C(=O)CCc1ccccn1 c1(-c2scc(OC)c2)cccc(S(=O)(=O)N2CCCCC2C(=O)O)c1 n1(C(C(=O)NCCC(C)N(C)C(C2CC=CCO2)=O)C2CC2)cc(Br)cn1 n1(CC)cc(Br)c(C(=O)NCC(C)N(C(=O)C(C(C)C)n2cnnc2)C)n1 C(=O)(C(C)(C)Cc1cnn[nH]1)N1CCC(C)C1.C1(C2(NC(=O)COC)CC2)CCOC1 Nc1ccc(C(F)(F)F)nc1C(=O)NCCN(C(=O)Cc1ccncc1)C1CC1 c1(C(=O)NCC2(OC)CN(C(C(CC)C)=O)C2)cnc2nc(Cl)ccc2c1 CCCCC(CC)CC(CC)Nc1ccc(NC(C)=O)nc1 C(=O)(CCCC(C)=O)NCCN(C(=O)Cc1cccc(OC)c1)CCC n1(CC)ncc(CN2CCC2C(=O)N(C2CCOCC2)C(C)C)n1 c1(NCC2(C(N)=O)CC2)[nH]c(=NC2COCC2N2CCOCC2)nc2scnc12 CC1CC(NC(c2ccc(C(F)(F)F)s2)=O)CN1C(c1ccnnc1S)=O c1(C(=O)NC2CCC(CCNC(C=CCC)=O)C2)ccc(NS(C)(=O)=O)nc1 C(=O)(C1=CCC(C)(C)CC1)N1CC(C(=O)NCC(CC(=O)NC)C)OCC1 c1(C(N2CC(C(=O)Nc3ncc(C)cc3C)C2)=O)cc(Cl)nc(Cl)c1F N1(C(Cn2c(C)nnn2)=O)CCCC12CCN(C(=O)C1=CC3CCCC13)CC2 C1(NC(c2cnc(CC(C)C)[nH]2)=O)CN(C(=O)Cc2ccnnc2O)CC12CC2 N1(C(c2c(CC)cco2)=O)CCC(CC)C1C(=O)N(CCS(C)(=O)=O)C Cc1ccc(C(=O)N(CC(C)NC(=O)CCC2OCCO2)C)c(C(C)C)n1 C12(C(=O)NCCN(C(C=C(C)Cl)=O)CC3CCCC3)CCC(COC)(C1)OC2 N1(C(c2n[nH]c(C)c2O)=O)CCC(C)CC1C(=O)NC1(c2nc[nH]n2)CC1 n1(-c2cn(C)nc2)nc(-c2cncs2)nc1-c1csc(-c2ccc(Br)cc2)n1 C(=O)(C(CC(C)C)NC(=O)C(O)C(F)(F)F)NCCN(CCC)CC c1(C(=O)NCC(CCCC)NC(c2c(Cl)noc2C)=O)ccc(C(C)=O)c(C)c1 C=CCC(CC)C(=O)N1CC(CCNC(C23CCC(CC2)CC3)=O)C(C)C1 c1(C(N(C)CC2CN(C(C3CC=CCC3)=O)CCO2)=O)cnc2occc2c1 C1(C(=O)NC(C2(C(N3CCC(N=[N+]=[N-])C3)=O)CC2)C)CCC2(CCC2)O1 CC1CCN(C(c2nccn3ccnc23)=O)CCN1C(=O)CCc1cn(C)cn1 C(=O)(C1=CCOCC1)NC(C1(O)CN(C(=O)Cc2nc[nH]n2)C1)C c1(OC)ccc(C(=O)NC2CC(NC(=O)CC(F)F)C23CCC3)cc1S(N)(=O)=O N1(C(=O)NCC(C(=O)OC(C)C)N(C)C)CCC2(CCC2)C(O)C1 N1(C(COCCCC)=O)CCC(CCNC(C2(C)CCOCC2)=O)CC1 c1(C(=O)NC2C(C)CN(C(c3ccc(Cl)cn3)=O)CC2)cc2ncccn2n1 c1(C(=O)NCC2N(C(COCC(=C)C)=O)CCC2C)cccc(C#CC2CC2)c1 CCCC(CC)C(=O)N1CC(C(=O)Nc2ccc(OC)cc2)C(F)(F)C1 C1(NC(c2onc(CC)c2C)=O)CCN(C(c2ccnn2C(C)C)=O)CC1CO C(=O)(CC(CNC(C)=O)CC(C)C)NCCCCN(C(CC(C)SC)=O)C C1(N(C(c2nccs2)=O)CC)CCN(C(c2occc2C(C)C)=O)C1 CC(CO)C(=O)NCC1CC(F)(CNC(C2(C3(C)OCCO3)CC2)=O)C1 Cc1ccc(N(C)C(C2CC(C)CN2C(C2CCC2C)=O)=O)c(C)c1 C1(C(=O)NCCOCCC(C)C)CCN(C(C2CCCS2)=O)C1 C(CN=c1[nH]c(NC2CCCCC2S(C)(=O)=O)nc2ccsc12)N(CCCC)C C(=O)(CC1OCCc2ccsc21)N(CCNC(C(C)(CO)OC)=O)C c1(CC(=O)NCC2C3CC2N(C(=O)C2=C(Cl)CCCC2)C3)n[nH]c2c1CCCC2 c1(CN(C(CNC(CC)=O)=O)C)ccccc1CNC(c1ccc(Cl)o1)=O N1(C(C(CCCC)CC)=O)CCC2(CC1)CN(C(=O)C(F)C1CCC1)C2 n1(CC(N2CCC(C(N(c3ccccc3)C)=O)C2)=O)ccccc1=O CC(CC(C)(F)F)C(=O)NC1(C2CN(C(=O)CC3COC(=O)C3)C2)CC1 c1(NC(C2N(Cc3[nH]c(C)c(C(=O)O)c3C)CCSC2)=O)ccnc([N+](=O)[O-])c1 Cc1cc(Cl)ncc1CN1CC2C(C1)N2C(C1CCCCC1(C)C)=O C(=O)(C(C(C)C)c1noc(C2CC2)n1)N(CCC)CC1(C)OCCO1 c1(C(N2CC(NC(c3c(I)ccnc3Cl)=O)C(F)C2)=O)nc2ccccc2[nH]1 C1(NC(CC(C=C)CC)=O)CCN(C(=O)C(c2cc(F)cc(F)c2)O)CC1(C)C N(C1CN(C(c2ccno2)=O)CCc2ccccc21)C(c1c(F)ccnc1F)=O c1(CC2(NC(C3C(CNC(COCC#C)=O)C3)=O)CC2)ccsc1 c1(OCC)c(F)c(C(N2CC(C)(NC(c3scc(C)c3Cl)=O)C2)=O)cc(F)c1F N1(CC)CCC(NC(C2COCCC2NC(=O)C(OC)OC)=O)C1=O n1(CC(C)C)cc(C(=O)NCCCN(C(=O)CC(C)N(C)C)C)cn1 c1(C(=O)NCCOc2ccc(Cl)c(Cl)c2)c[nH]c2c(Br)cccc2c1=O c1(C(N2C3(CN(C(c4cc(CC)[nH]n4)=O)C3)CC2)=O)cc(C)cc(Br)c1N c1(C(=O)NCC=C2CCN(C(C3CC(C)C3)=O)CC2)cnc2ccoc2c1 C(C(C(C)(C)C)NC(=O)CCc1cccs1)NC(COCCCC)=O C1(C(=O)NC2CC(C)(NC(c3nc(COC)sc3)=O)C2)CCCCC12CCC2 C#Cc1cc(F)c(C(N2CC(NC(C3(C)CC(F)C3)=O)C(C)C2)=O)c(F)c1 c12cn(nn1)Cc1nc(cs1)NC(=O)C2.C1(N2CCCC2)CCC1CC1CCC1 Cc1c(C(N2CC(NC(c3cncn3C)=O)CC(F)C2)=O)cc(F)cc1[N+](=O)[O-] c1(OC)ncc(NC(C2CC(C(=O)O)C23CC3)=O)c(C)n1 C1(NC(C(COC)O)=O)CCN(C(c2ccc([N+](=O)[O-])[nH]2)=O)C1(C)C C(C)(C)(CC(=O)NCCSCC(=O)NC1C(C)C1C)OC C=C(F)C1(CC(N2CCCCC2CCC(N2CC(CC)(CO)C2)=O)=O)CCC1 C(=O)(C1=C(Cl)CCC1)NC1CN(C(c2c(C(=O)OCC)con2)=O)CC1O c1(C(=O)NCC(C)(C(C)C)NC(CC(CCC)C)=O)noc2ccc(Cl)cc12 Fc1ccc(C(c2nnnn2C2CC2)NC2CC(C3CCC3)C2)cc1C(F)(F)F CC1CN(C(C2CCC3(CC3)N2C(=O)CC2CCC=CCC2)=O)CC(C)(C)O1 C1(F)(CNC(c2cc(Cl)nnc2O)=O)CCN(C(C2(CC(F)(F)F)CC2)=O)CC1 c1(OC)nc(C(=O)NC23CCN(C(=O)Cc4noc(C)c4C#N)CC2C3)ncc1F CC1(C)CCC(C(=O)NC2CCN(CCCNC(c3cc[n+]([O-])cc3)=O)C2)C1 c1(CC(=O)NC(CC(C)C)CNC(=O)C(C(C)C)N(C)C)cccc(Cl)c1Cl C1(O)(C(N2CC(OCCNC(C(C=C)O)=O)C2)=O)CC2CCC1C2 c1(OCC#C)ncccc1C(=O)NCC(C(C)C)NC(C1CC1C(F)(F)F)=O Cc1ncccc1CC(N1CCC(CNC(=O)CC2COC(=O)C2)C1C(C)C)=O N1(C(C(COCC)NC(=O)C(C(C)C)SCCOC)=O)CC2CSCC(C2)C1 c1(C(=O)NC2CC(NCc3cnc(C4CC4)s3)C2)cnc(O)c(Br)c1 c1(C(N(CC(CN(C(C(C)NC(CC)=O)=O)C)O)C)=O)cnc(N)cn1 C1(CNC(c2c[nH]nc2[N+](=O)[O-])=O)C(O)C(O)CN1C(=O)COCC1CCCO1 CC1CN(C(c2ncc(-c3ccc(C4CC4)nc3)cn2)=O)CC(C)O1 C(=O)(C1CCOc2ccccc21)NCC(CC)NC(=O)CN(CC(C)(C)C)C C(=O)(CCCCC(=O)N1CSCC1C(=O)NC(CO)CCC1CC1)OC c1(OC)ccc2c(c1)C(NCc1cnc(C)cn1)CCCO2 CC1CN(C(c2csc(C#N)c2)=O)CC1NC(=O)C(c1ccc(Cl)nc1)(F)F C1(NC(CC2(C=C)CN(C(=O)CCc3cncn3C)C2)=O)CCC2(CCC2)C1 Cc1cccc(C(C)CNC(N2CCCC(O)C2)=O)c1 CC1CN(C(c2cc(Cl)ccc2Cl)=O)CCC1N(C(=O)CCCF)C N1(C2CC3(CC(O)(C(F)(F)F)C3)C2)CCn2c(cnc2-c2ccccc2)C1 c1(OCC)ncccc1C(N1CC(C)(NC(c2conc2C)=O)C1)=O C1(CN(C(COCC#C)=O)C)CCN(C(=O)CC(C)c2cccnc2)C1 CC#CCCC(=O)Nn1ccccc1=O.C12CCCCN1CCc1cn(nn1)C2 Cc1ccc(F)cc1C(=O)NCC1CN(C(C2CCC(=O)N2)=O)CC1C N1(C(C2CC2c2ccncc2)=O)CCCC(O)(CCNC(C2CCSCC2)=O)C1 C1(C(=O)NCC2N(C(c3c(OC)csc3)=O)CC(OC)C2)CC2C(C1)C2(F)F C1(C(N2CCC(CNC(C(C)OCCN(C)C)=O)CC2)=O)CCN2CCCC2C1 Cc1cc(N(C)CCc2nccc(O)n2)nc(=NCc2nc(C(C)C)cs2)[nH]1 Cc1ccc(C(=O)NCCC2CN(C(C3(n4cncn4)CC3)=O)CCO2)nc1 c1(C(C)=O)cn(CC(C)(C)CNC(C2CCCCO2)=O)nn1 N1(C(c2cn(C)nn2)=O)CCCC(CO)(NC(=O)C2=NOC(c3ccccc3)C2)C1 c1(C(=O)OC)cc2c(NCCC(CC)(CC)NC(c3cnsc3)=O)ncnc2[nH]1 c1(C(=O)OC)cc(C)cnc1N1CC(CO)(NC(=O)CC2CC(O)C23CCC3)C1 N1(CCc2cn(Cc3c(OC)c(OC)c(Br)cc3)nn2)CCCC2(CCCO2)C1 c1(C(=O)NC(CCNC(C2(OC)CCCCC2)=O)C)cccc(C(C)C)c1F c1(C(N2CC3C(NC(c4c(N(C)C)cccn4)=O)C3C2)=O)ccc(O)c(F)c1F C1(C(=O)NC2CCCN(C(C=Cc3nc(C)sc3)=O)C2)CCC(C)(C)CC1 C(CCC(=O)N(C(C)CNC(=O)CC1(C)CCCC1)CC)NC(=O)OCC C1(C(N2CC(C)SCC2)=O)CC(F)CCN1C(=O)C(CO)N(C)C N1(C(C(CN(CC)CC)F)=O)CCC2(CC(NC(C3(C)CCC(=O)N3)=O)C2)C1 c1(N(C(c2cc(C)c(Cl)c(N)c2)=O)C)ncnc2sc(Br)cc12 N1(c2nccc(C)n2)CC(C(=O)NCc2nc(Cl)ccc2F)OC2(CCC2)C1 CN1C(=O)COCC1CNC(C1CCCN(C(=O)C(F)C2CCCC2)CC1)=O c1(C(N2CCC(OC)C23CCC3)C(=O)NCCOC)ccc2cc(F)ccc2n1 N1(C(C2(C)COCCO2)=O)CCCC12CCN(C(=O)CC1CCCCCO1)CC2 CC1(C)COC(C(N2CC(O)(C(C)(C)CNC(c3cc(Cl)cs3)=O)C2)=O)C1 N1(C(CC=CC)=O)CCCC(CC)(NC(c2[nH]nnc2CC)=O)C1 CN1CCc2c(C(=O)NC3CCN(Cc4cccc(C#N)n4)C3)cccc21 CC(C)CS(=O)(=O)CCC(=O)N1CCCC(CN(C(=O)C(=O)N(C)C)C)C1 C1(C(N2CCC2C2CCC2)=O)C2CCCC2CN1C(=O)CC1CSC1 c1(C(=O)NCC=CCNC(c2cccnn2)=O)ccc(Cl)c(Br)c1 c1(OCC(=O)NC(C)(CNC(C23CC(O)C2C3)=O)C2CC2)c(F)cccc1F C(=O)(CC1COc2ccccc21)NC(C)CCNC(c1c[nH]nc1F)=O C1(NC(C(C(C)C)C)=O)CCCCN(C(=O)CCOc2ccccc2)CC1 CC(CCC(=O)NC1CC(Cl)(Cl)C1)NC(=O)Cc1cc[nH]n1 C1(NC(c2cc(CC)sn2)=O)CN(C(C2C3(CCC3)C23CCC3)=O)CC1C1CC1 c1(C(=O)NCC(C2(O)CCN(C(C3(CO)COC3)=O)C2)C)cncc(C2CC2)c1 CN1C(=O)CCCC1C(=O)Nc1cccc(CC(=O)C2CC2)c1 c1(C(=O)NCC=CCNC(C2CC2CN2CC(CO)C2)=O)cc2ccc(Cl)cc2[nH]1 C1(F)(CNC(c2cccc(Cl)c2)=O)CCCN(C(C2CCOC2C2CC2)=O)C1 c1(C(=O)NCC(CC)NC(=O)CC2CC=CCC2)cc(F)c(C#N)c(F)c1 C(CCC(C)C)(C(=O)NC(C)Cc1nn[nH]n1)NC(CNC(=O)OC)=O C1(CNC(c2occc2F)=O)CC2(CCN(C(=O)CC3(O)CCCCC3)C2)CO1 C=CCC(C)(CC)C(=O)NC1CC(C(C)NC(=O)CCC(CF)CF)C1 C1(C(C)=O)C2C3CC4C1C1C2CC3C41.N12CC3(CC(CO3)NC1=O)C2 CC(C)CC(C)C(=O)N(C)CC1CCCCN1C(=O)CCCN1C(=O)CCC1=O c1(C(=O)NCC2CCN(c3nccc(C(F)F)n3)CC2)cc(F)c(F)cc1Cl N1(C(CN(CCC)C)=O)CC(C(=O)NCCCC(F)F)CCC1(C)C C(=O)(CC(O)C(C)C)N1CCC(c2cc(CNC(CC3(C=C)CC3)=O)on2)CC1 c1(C2N(C(c3cc(C)ns3)C(=O)NCCC3CC3)CC2)ccc(Cl)c(Cl)c1 N1(C(C(=O)NC)=O)CC2CN(C(=O)C=CC(c3ccc(C)cc3)=O)C2C1 N12CCC(C)C(C1)N(C)C(=O)C2=O.c1(NC(=O)CCC#N)ccc(OCCF)cc1 C1(C(=O)OCC)COC2(CNC(=O)C(O)c3ccco3)CC1C2 CCC(CC(=O)N1CCC(C(=O)NCc2nn[nH]c2C2CC2)(CO)C1)C(F)F c1(C(=O)NC(C2CCCCC2)CNC(C2(CCCC)CC2)=O)cc(C#N)c[nH]1 c1(OC)cccc(C(N2CCCC2C(=O)NCC(C)(C)C2CC2)=O)n1 C#Cc1ccc(CNC2CN(C(COC(=O)C(C)OCOC)=O)C2)cc1 C12(C(=O)NC(C3CCOC3)CNC(C=Cc3cc(C)no3)=O)CC(C)(CCO1)C2 c1(OCC(=C)C)ccccc1C(N1CCC(NC(C2(F)CCOC2)=O)CC1)=O c1(C(=O)NCC(CC(C)C)NC(c2ccc(CC)s2)=O)nn(C)c(C)c1Cl n1(CC(=O)NC(C2(CNC(C=C(C)C)=O)CC2)C)cnc(C#N)n1 c1(C(N2CC(OC)C(NC(c3cc(Cl)cs3)=O)C2)=O)ncc(C)cc1F C1(C(=O)NCc2ncc(C)o2)CCCCN(C(=O)C(c2cccc(Cl)c2)(C)C)C1 c1(CN2CCOCC(NC(Cc3c(OC)cccc3)=O)C2)cc(Cl)c(O)c(Br)c1 N1(C(C(C)C2(O)CCC2)=O)CC(C(=O)Nc2cncc(CO)c2)CC(C)(C)C1 c1(C(=O)NC2CN(C(c3nc(Br)cs3)=O)CC2F)ccncc1F CCC(=O)CCC(=O)N(CC(=O)N(C)Cc1cccc(O)c1)C1CC1 c1(SC(C)C(=O)NC23CC(C2)N(C(=O)C2=CCCS2)C3)ccc(F)cc1 c1(CCC)ocnc1CNC(=O)Nc1cnn(CCCOCC)c1 N1(C(C2(CC(C)C)COC2)=O)CC=CC(NC(=O)C2=C(C)CC2)C1 C(=O)(CCCCC#N)NC(C(=O)NC(C#C)CC1CC1)(C)C1CCC1 CCN=c1[nH]cc(C(=O)NCCCCN2CCCCC2)s1 Cc1cscc1C(=O)NC(CN(C(=O)CC1(C)CCCC1)C)Cc1ccccc1 C1(C(=O)NC23CC(NC(CC4CCC(C#N)C4)=O)(C2)C3)CCc2ncnn2C1 C(=O)(CC(C)CC(C)(C)C)NC1(CC)CCN(C(c2cc(C)nnc2O)=O)CC1 C(=O)(C(CCC1CC1)N(C)CC1CCCCC1)NCCSC c1(CNC(=O)CCC2CCOC2)cccc(NC(C2C=CC(CF)C2)=O)c1 c1(CC2C(=O)N2)cnn(C)c1O.N1(CCNC(C(=O)NCC)=O)CCNC1=O C(=O)(C(C)(CO)NC(c1ccnnc1O)=O)N1CC(c2nc(C)[nH]n2)C1 c1(C(=O)NCCC2(CNC(C(N3CCC(C)C3)=O)=O)CC2)cnn2ncccc12 c1(C(=O)NC2CN(C(C(C)=CC)=O)CC2CC(C)(C)C)cnn2c1C(C)CCC2 c1(C(N(C(C)CCNC(c2cnoc2C2CC2)=O)C)=O)cc(F)cc2nn[nH]c12 N1(C(c2cc(CNC(c3ccncc3F)=O)sc2)=O)CC2C=CC2C1 C1(C)(C(N(CC(CC)NC(c2ccoc2Cl)=O)C)=O)CCN(C)C1=O CC(C(=O)NCC1CN(C)CCN1C(C1(Oc2ccccc2)CC1)=O)C(C)(F)F CCCCCC(C(=O)NC(C)CCCCNC(c1ccn(C2CC2)n1)=O)C(C)C CC1CN(C(C2CCSC2)=O)CC(C)N(C(C2CCCC2(C)C)=O)C1 N1(C(C(C)CC2CC2)=O)CCC(C(C)CNC(c2cnc(N(C)C)nc2)=O)CC1 c1(C(CN(C)C(=O)NCCCNC(c2ccccc2)O)O)ccc(O)cc1 c1(OC)cc(C(=O)NCC#CCNC(=O)CS(=O)(=O)CCO)cc([N+](=O)[O-])c1Cl C12(NC(C3C(C)C3C)=O)CCCC1N(C(=O)CC1(O)CCOC1)CCC2 C(N=c1[nH]cncc1Br)C1C(C)CN(C(c2cc(Cl)ccc2Cl)=O)C1 c1(C(=O)NC2CC(NC(C3(CC#C)CCC3)=O)C2)cc(Cl)no1 N1(C(C2C=C(C)CS2)=O)CC(C(=O)NC(C)(C)C(C)(C)C)CC(C)(C)C1 C(=O)(C1=CN2CCS(=O)(=O)N=C2C=C1)N1C2CN(C(CCS(C)=O)=O)C(CC2)C1 C1(C(N2CCCCC2)=O)CC2CCCCC2N1C(=O)CCNC1COC1 Cc1ccc(C)c(CNC(C2C3CC4C(C3NC(c3coc(CO)c3)=O)C24)=O)c1 C1(C(N(CC(CC)NC(CCOCC)=O)C)=O)CS(=O)(=O)CC12CC2 c1(NC(C2CC3CC3N2c2ncc(Br)cn2)=O)nccc2cccnc12 N1(C(COC)=O)CCCC1CN(C(=O)Cc1cnoc1)C C1(CNC(c2ccoc2Cl)=O)C2CCCC1N(C(=O)Cc1ccc(F)cc1F)C2 c1(C(N2CC(F)CC(NC(c3n(CCC)ccc3)=O)C2)=O)c(F)cc(O)cc1F CC1CC(CNC(=O)C(F)(F)c2cncs2)CN1C(c1cccc(C2CC2)c1)=O c1(NCC(C)(C)NC(CN(C)CCO)=O)cnc(C#N)cn1 C(=O)(C(C)C(O)C(C)C)NC(C(=O)N(CC(C(C)C)OC)C)CO c1(C(N(C2CCC(NC(C3(C(F)(F)F)CCC3)=O)C2)C)=O)cccc2nccn12 c1(CC)ccc(C(N2CC3CC2CC3NC(c2cc(C3CC3)cs2)=O)=O)cc1F N1(CC(=O)NCc2ccccn2)CCCC1C1OCCO1 c1(C(N(CCCOCCN(C(C(CC#C)C)=O)C)C)=O)cnn2cccc(Cl)c12 N1(C(C(C(C)C)NC(=O)N(C)C)=O)CCC2(CC1)CC(OC(=O)C(F)(F)F)CO2 CC(C(=O)N(CCCCN(C)C(C1CC2(CCOC2)C1)=O)C)C(F)(F)C(F)F C(CN=c1[nH]c(=NCCCF)c2cccc(F)c2[nH]1)SC(C)C C(c1ccccc1F)=CC(=O)NC(C)CC1CCN(C(C2CC23CCOC3)=O)CC1 c1(C(N2CCC(NC(COCCSC)=O)C2)=O)c(C)oc(C)c1S(N)(=O)=O c1(C(=O)NC2C3CN(c4nc(CC)cc(CC)n4)CC32)c2c(nn1C)CCSC2 c1(-c2n(C)nc(-c3cccnc3O)n2)cc2cc(Cl)ccc2n1C c1(C(=O)NC2(C3CCCN3C(C3CC4(CC4)CO3)=O)CC2)cnc2[nH]nnc2c1 CCCCC(CNC(=O)C(CCC)NC(N)=O)NC(c1cc(C(N)=O)c[nH]1)=O c1(CC)nn(C)c(C(N2CCC(COC)(NC(=O)C(N)=O)CC2)=O)c1Cl c1(C(=O)NC2(CC=C)CCN(C(C3CC4(CC4)CO3)=O)C2)c(C=C)cnn1C c1(OC)cc(C(N2CCCC2C(C)(C)O)=O)ccc1F Cc1nc(C(C)(C)C)ncc1C(=O)NC1CC(CNC(=O)C(C)(C)C)C1 c1(C(N2CCC(CN(C(=O)C(C)N3CCCC3)CC)CC2)=O)c(N)cccc1F C=CC(C)CC(=O)NCCC(C)NC(c1csc(Br)c1C)=O C1(OC)CC(CNC(c2[nH]cnc2C#N)=O)N(C(C2CCCN2C)=O)C1 Cc1cn2c(C(=O)NCC3CC4COCC4N3C(=O)C#CC3CC3)cnc2s1 C1(CCC(=O)NCC2CCN(C(=O)CC3CCCCO3)C2)CCC(O)CC1 CC1(C)C=C(C(=O)NCCCC2CN(C(=O)C(c3ccc(F)cc3)F)CCO2)C1 N1(C(CNC(C=C)=O)=O)CC2CN(Cc3c(F)cc(F)cc3F)CC2C1 c1(C(N(C)CC2CCCN2C(=O)C=C(Cl)Cl)=O)ccc(Cl)c(Cl)c1O C(=O)(CCC(CF)CF)NCCC12C(CN(C(Cc3nc(CC)sc3)=O)C1)CC2 c1(C(=O)NCC(CC)NC(c2n[nH]c(C)c2C)=O)ccc2ncnn2c1 C(=O)(C1=CCCSC1)N(C1(C(=O)NCC2C(C)(C)COC2)CCC1)C1CC1 C(CC(C)C)(C(=O)N1CCC(C(C)(C)C(N2CCC(O)(CO)CC2)=O)C1)OC c1(OC)cc(C(=O)NCC2CCC(NC(=O)CC3CC34CC4)CC2)cc(OC)n1 c1(C(=O)OC)cc2[nH]c(C(=O)NCc3[nH]c(C)c(C(=O)O)c3C)cc2s1 C=CCC(C)(C(=O)NC1CCN(C(=O)COc2ccc(F)cc2)CC1C)N(C)C N1(C(Cc2c(C)occ2)=O)CC2(CCN(C(c3cn4c(n3)CCCC4)=O)CC2)C1 C(C(F)(F)C(F)(F)C(F)(F)C(F)(F)F)NC(CC(C)Cc1ccc(Cl)cc1)=O C1(NC(c2nc(C)sc2)=O)CN(C(C2CN(C3CCOC3)C2)=O)CCC12CCC2 C(=O)(C(C(=O)NC1(CO)CN(C(=O)C(C)NC(=O)COC)C1)C(C)C)OCC C1(C(=O)NCCN(C(C2N(C(C)=O)CCC2)=O)C2CC2)CCn2nnnc2C1 Cc1cc(F)c(C(N2CCC(N(CCO)C(c3ccc(C#N)o3)=O)C2)=O)cc1F CC1CN(C(C2CCCN2C=O)=O)CCCN1C(=O)C=CC1CCC1 CCCCCCC(CC)C(=O)N1CCCC1CN(C(=O)CCCCC(=O)NC)C c1(C(=O)NCCOCCN(C(C=CC(C)(C)SC)=O)C)ccc2cn(C)nc2c1 c1(-n2cc(C(CC(N)=O)NC(C3(C=C)CC3)=O)nn2)cccnc1Cl N1(C(COC(C)(C)C(F)(F)F)=O)CCN(C(C2CCCO2)=O)CC1C1CCC1 Cc1nc(CN2CCN(C(=O)CC(=O)N(C)C)CC2)cc(=NCC2CC2)[nH]1 c1(C(N2C(CN(C(c3ccc(C)n3C)=O)CC)CCC2)=O)ccc(C)c(C)c1 CC1CC(C(C(=O)NCC2CCOC2)N(C)Cc2cocn2)CC(C)C1 CC1=C(C)CN(C(=O)CN(C)C(C2COCC(C)O2)=O)C1 N1(C(c2cc(OC)no2)=O)CCC2CN(C(c3ccc(NC=O)cc3)=O)CC2C1 N1(C(CC2CC(=C)C2)=O)CCOCC1Cc1cn(CC2CCC(=O)O2)nn1 c1(CN2CC(NC(=O)CCc3ccsc3)C(F)C2)cc(Cl)c(F)c(Cl)c1 C12(NC(c3nc(OCC)sn3)=O)CCCC1CN(C(=O)C=Cc1cccs1)C2 C1(NC(CC=CCC)=O)CCOC(C2CCN(C(=O)COCC(C)(C)C)CC2)C1 C1(C)(CNC(CC2C3CN(C(CC4CC(OCC)C4)=O)CC32)=O)CCC(O)CC1 CC1CN(C)C(C)CC1NC(C1(C)C=CCN1C(=O)CC1CC(N(C)C)C1)=O c1(C(N2CCCC(C(O)C(F)F)C2)C(=O)NC(CC)C)cnc(OC)c(F)c1 N1(C(c2ccc(CC)o2)=O)CCCC(CO)(CNC(=O)COc2ccon2)C1 c1(C(N2CC(CNC(C3CC(OC)C(OC)C3)=O)OCC2)=O)cnc(Cl)c(N)c1 N1(C(CCc2cc(C)nn2C)=O)CC(NC(=O)C2=CCCSC2)C2(CC2)C1 N1(C(c2cc(C)c(Cl)cc2)=O)CC2CCC1C(NC(=O)C=C1CCC(C)CC1)C2 N1(C(C(C)OCC)=O)Cc2[nH]nc(C(=O)NCc3ccn(CC)n3)c2C1 C1(C(N2CCC(NC(C(C)(C)SC)=O)CC2)=O)CC2OC(C)(C)OC2C1 C1(CC(=O)NCC(C)NC(=O)CCCN2CCCCC2)OCCCO1 c1(C(=O)NC(C(C)NC(=O)CC23COC(C)(C2)C3)C)ccc2ccn(C)c2c1 C1(C#CC(=O)NC(CCN(C(=O)C(C)(C)C(C)C)C)C(C)C)(CC)COC1 c1(CN(CC)Cc2ccc(C)cc2)cn2c(n1)CCN(CCn1cccn1)CC2 CCC(CNC(=O)CN(C1CC1)C(C)C)(CC)C(=O)N1CCN(C2CCC2)CC1 C1(NC(CCCOC(C)C)=O)CN(C(C2(O)CC2(C)C)=O)CC2(CCC2)C1 C(C(C(=O)N(CC(O)CC)C)NC(c1cc(C(C)C)[nH]n1)=O)OCC CC1(C)CCC2(CC1)CC2C(N1CC(NC(c2cnn3cc[nH]c23)=O)C1)=O CC1CN(C(c2cncc(N)c2)=O)CC1CCNC(C1CC(=O)N(O)C1)=O CCCCC(C)CCC(=O)N1CCCC1CN(C(=O)C(c1ccc(C)o1)C)C c1(OC)cc(CO)c2c(c1)CCC2.c12ccnc(c1)CCn1cc-2nn1 c1(SC(C)C)ccccc1C(=O)NC1CC(C)N(C(c2ncc[nH]c2=O)=O)C1 c1(NC2CN(C(Cc3nc(C)sc3C)=O)CC2C)ncnc2cc(F)ccc12 C1(C(N2CC3CCN(C(=O)C4CC4)C(C3)C2)=O)CC12CCOc1ccccc12 c1(OC)cccc(S(=O)(=O)N2CCOCC2CNC(=O)CC2CC2)c1 C(=O)(CC(C)CNC(=O)C(C1CCCO1)NC(c1cnc(C(C)C)o1)=O)NC C(C(F)(C(=O)N1CC(C)(C(F)(F)F)C1)C(C)C)NC(COCC#C)=O N1(C(C=C(CC)C)=O)CCCC1C(C)NC(=O)C(C)(C)c1ccccn1 C(N=c1ccnc[nH]1)C1CCN(C(c2cccnc2C2CCCC2)=O)C1 N1(C(C2(CN(C)C)CC(=C)C2)=O)CCC(N2CCOCC2)CC1 CC1(C)CC(=O)CCC1C(=O)NCC(CO)NC(C1CCC(=O)N1)=O C1(NC(C2OCCC(NC(c3occ(C)c3)=O)C2)=O)CCCCCCC1O c1(CC(C(=O)NCCCNC(CCc2onc(CC)n2)=O)C)cccc(F)c1 C(C)(CC(=O)NC(C)Cn1cc(CC(O)C2CC2)nn1)OC C1(CNC(C(CC#C)O)=O)CCN(C(c2cnn(C)c2Br)=O)CC1O c1(C(N2CCC(C(C)NC(c3cnc(OCC)s3)=O)C2)=O)ncc(Cl)cc1Cl C=CCCCC(=O)NC(c1ccc(C(C)C)cc1)CNC(=O)CO CC1c2cc(F)ccc2CCN1C(c1cc(Cl)cc(Cl)n1)C(=O)NC1CCCC1 C1(N(C(=O)Cn2cc(C3CCC3)nn2)CC)CCCN(C(=O)Cc2nc[nH]n2)C1 C1(CC#C)(C(=O)NCCSCCCO)CCN(C(=O)C=CCCC(C)C)C1 C1(C(=O)NCCN=[N+]=[N-])CCC2CCC1N2C(C1(N2CCCC2)CC1)=O C1(C(=O)NCCOCCN(C(c2cc(CC(C)C)[nH]n2)=O)C)CCCCC1C C1(C(N(C(C)CNC(c2ccnc(-n3cncn3)c2)=O)C)=O)CC1C1CCCC1 C1(OC)COCCC1CC(=O)NCC1(NC(=O)CCC(C)O)CCC1 C1(NC(c2ccc(C)cc2C)=O)CCCCCN(C(c2cn(C)c(O)n2)=O)C1 C1(C)(NC(c2cnc(C)[nH]2)=O)CCC(NC(=O)Cn2ccc(C3CC3)n2)CC1 C(=O)(CC(C)C(F)(F)F)NCC(C)NC(=O)Cc1cnccc1C(F)(F)F CC(CC1CCC1)N=c1[nH]c(=NCc2ccc(Cl)o2)[nH]c2c1CSC2 O=C1CSc2ccc(C(=O)NC3CN(C(=O)Cc4cnsc4)C4CC34)cc2N1 C12(COC)COC(C(N3CC(C)(NC(C4COC(=O)C4)=O)C3)=O)(C1)C2 C=C1CC(C)(C(=O)NC2CCC2CNC(=O)Cc2cnc(C)s2)C1 C1(CNC(c2c(CC)cco2)=O)CC(C)N(C(=O)COC(C)(C)C)C1 c1(C(=O)NCCNC(c2cc(C(N)=O)[nH]c2)=O)ccc(S(=O)(=O)C2CC2)cc1 CC1CCC(C(=O)Nc2cccc(CF)c2)N1C(c1cccc(C(F)(F)F)c1)=O CC1CC(N(C)C)CN(C(N2CCCCC2C(=O)OC)=O)C1.N1(CC)CCCC1 C(C)(C)(CN=c1[nH]c(N2CCC(CO)C(C)C2)nc2c1CSC2)OC(C)C c1(C(N2CCC(N(C(C=CS(C)=O)=O)CCO)C2)=O)ccc2ccccc2c1F c1(C(=O)NC(CNC(C=Cc2cnc(C)s2)=O)CC(C)C)cnc2ccnn2c1 C(=O)(CC(C)(O)C(F)(F)F)N1CCC(C(C)NC(=O)CCc2ccc(O)nc2)C1 C1(N(CCNC(C)=O)C(c2csnc2C)=O)CCN(C2CCSC2)CC1 CC1CC(CNC(C2CC(F)(CO)C2)=O)CN1C(c1cc(F)c[nH]1)=O c1(C(N(CCCNC(C2C(=C)C2)=O)C)=O)csc(C2CCCO2)n1 N(S(=O)(=O)N1CCC(CC(=O)O)C1)CCO.C=CCO C1(CNC(CN(CC)CC)=O)CCC(NC(C2CCNC(=O)C2)=O)CC1 c1(-c2ccc(CNC(c3cccc(N(C)C)c3)=O)cn2)ccc2sccc2c1 N1(C(c2c(N)nccn2)=O)CC2CC(NC(c3ccnnc3)=O)C(C2)C1 C1(C(N(C2CCN(C(c3cccc(C4CC4)c3)=O)C2)C)=O)CCCC1(F)F N1(C(=O)CC2CCCO2)CC2CC2(C(N2CC(O)(c3cc[nH]n3)C2)=O)C1 N#Cc1ccc(C=CC(=O)NC2CC3CCC2(NC(=O)CN2CC=CC2)C3)cc1 Cn1cc([N+](=O)[O-])cc1C(N1CCC(NC(=O)CC2CCCCC2O)C(F)C1)=O C1(CC)CN(C(c2ccc(=O)n(CC)n2)=O)CCN1C(C1CCC(OC)C1)=O C(C)(C(C(=O)NCCc1nncs1)C(C)C)NC(c1c(C)n[nH]c1)=O c1(C(N2CCC(C(C)NC(CCc3ncc(C)[nH]3)=O)C2)=O)cc2sccc2s1 c1(OC)cc(C)c(CNC2CC2C(=O)Nc2nncs2)cn1 Cc1cc(C(=O)NC2CCCN(c3ccc(C#N)cc3)C2=O)cc2c1CCC2 C(=O)(C1=CC2(CCOCC2)C1)NCC(CC=C)NC(c1ccc(CO)o1)=O CCC(O)C(C)C(=O)N1CCC(C(=O)N(CC(C(C)C)OC)C)(CF)C1 N1(C(CC(C)N(C(c2ccoc2)=O)CC)=O)CCN(C(=O)C(C)SC)CC1 c1(CCC(=O)N(C2CN(C(=O)Cc3cc(C(F)(F)F)nn3C)C2)C)ccc(O)nc1 CC1(C(N2CCC(OC3CCOC3)C2)=O)CCCN(C(=O)CSC(F)F)C1 N1(C(C2(C)CC(=C)C2)=O)CCOC(CNC(=O)CCN(CC(C)C(C)C)C)C1 N(C1CN(C(c2cccs2)=O)Cc2ccccc21)C(C(CCC)(C)O)=O C(=O)(CN=S(C)(C)=O)NC(C)CN(C)C(C1CC1Sc1ccccc1F)=O c1(C(=O)NC2C(NC(C(C)NC(c3ccco3)=O)=O)C2)c(Cl)ccc2c[nH]nc12 C1(OC)CCC(C(=O)NCC(C)NC(=O)C(C)(C)OC(C)C)CC1 c1(C(C)NC(=O)C(N2CCC(OC3CCC3)C2)=O)ccccc1C1CCC1 Cc1cc(-c2nc(C(=O)NC(C)C(F)(F)F)c(C)s2)cnc1F N1(C(c2cnc(C)s2)=O)CC2C(NC(C3(C)CCC(=O)N3)=O)C2C1 C1(CNC(c2c(C)noc2)=O)(NC(C2CCN(CC(C)C)C2)=O)CCCCC1 C(CC(=O)N1CCC(C)(CNC(=O)C(CC(C)C)OC)CC1)(C(C)C)OCC C1(OC)CC2CC(C(=O)NC3(C(=O)NCC4CCN(C(N)=O)CC4)CCC3)CC12 C(=O)(C(CC(N)=O)NC(=O)C(O)C(F)(F)F)NCC1C(OCC)CC1 C1(C(=O)NCC(C)(C)NC(C2C(CC)C2)=O)(CF)CC(F)(F)C1 C1(CNC(c2cn(CCC)nn2)=O)CN(C(c2cnc(C(C)C)s2)=O)CCO1 Cc1[nH]c(C)c(C(=O)NCC2CC(C)N(C(c3sc(N(C)C)nc3Cl)=O)C2)c1C C1(O)(C(C)NC(c2ccn(CC)n2)=O)CCN(C(C2COC3COCC23)=O)CC1 c1(C(=O)NC2CCC(CNC(CC(C)O)=O)CC2)ccc2nn[nH]c2n1 N1(C(C=C(CC)C)=O)CCN(C(=O)CNc2ccccc2[N+](=O)[O-])C(C)CC1C C1(NC(C(CC)(F)F)=O)CC2CCC(C1)N2C(c1ccccc1OC(F)F)=O C(=O)(C(C)CC(C)(C)C)N1CCN(C(Cc2cc(CC)no2)=O)C(CCOC)C1 CC1CC(CNC(C2C=CCCC2)=O)CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)C1 N1(C(C2(NC(c3ncccc3F)=O)CCCC2)=O)CCCC(C2CCC2)C1 N1(C(C(c2cccc(O)c2)C)=O)CCCCC1CCNC(=O)CCc1cn[nH]c1 Cc1c(Br)csc1C(N1CCCCC1Cn1cc(-c2cccc(F)n2)nn1)=O c1(C(=O)NC(C2CN(C(C3CCS(=O)(=O)C(C)C3)=O)C2)C)noc2ncccc12 N1(C(C(F)OC)=O)C2CCC1CN(C(c1ccccc1O)=O)CC2 C1(CC(=O)NC(C)(CO)C2CC2)CN(C(C2CNC(=O)O2)=O)CCO1 N1(C(C(F)=C(C)C)=O)CC(NC(=O)Cn2cnnc2)CC(C)C1 C1(NC(C2(CO)CCCO2)=O)CCC2(CCNC2)C1 c1(C(=O)NCC(CNC(C(CC)NC(N)=O)=O)O)cc2scnc2[nH]1 CC(C)(CCC(=O)N1CCN(CCO)CC1)NC(=O)C=Cc1ccoc1 c1(CC)ccc(C(=O)NCC(C2CCOC2)NC(c2n[nH]cc2C(F)(F)F)=O)o1 c1(SCC(=O)NCCC(=C)CNC(=O)C(C)(F)CCCC)ccc(Cl)c([N+](=O)[O-])c1 c1(CCC(=O)NC2(C)CC(NC(C=C(CCC)C)=O)C2)cnc2n1CCCCC2 C12(C(=O)NC3(CNC(C4(c5cccc(C)c5)CC4)=O)CC3)CCCC1C2(F)F C#Cc1ccccc1CC(=O)NC(C1CN(c2cc(C(=O)OC)ncn2)C1)C C12COCCN1CC1(C3N(CCOC3)C2=O)CC1.n1(SC2CC2)cccn1 C(=O)(C1=NOC(C)(C)C1)NCC(c1ccc(F)cc1F)NC(C=CC(C)C)=O C1(C(N)=O)CCCN(C(C2CCC(CNC(=O)Nc3cnnn3C)C2)=O)C1 C=C(C(=O)N1CCOC(C(=O)Nc2cnc(Br)cc2C(N)=O)C1)C(F)(F)F N1(C(CC(C)NC(N)=O)=O)CCCCC1CN(C)C(c1cccc(N(C)C)c1)=O C(=O)(CCC(C(C)C)NC(C1(C)CCC1)=O)NCc1ccc(C)c(O)c1 Cc1cc(C)n(CCCNC(=O)C(=O)NCCC2CCCCO2)n1 CC(C)CC(C)(C)NC(c1ccncc1)C(=O)NCSc1ccccc1 CC1CN(C(c2cccnn2)=O)CC1CNC(C1(P(C)(C)=O)CC1)=O C1(NC(c2c(CC)cns2)=O)CS(=O)(=O)CC1NC(=O)CN1CCCOC1=O c1(OC(C(=O)NC(CN(C(C(CC)OC)=O)C)(C)C)C)ccc(Cl)cc1C C(C(C)C(=O)N(C)CC1CN(C(=O)CC2(n3ccnc3)CC2)C1)OC c1(C(=O)NCC(c2cc(F)cc(F)c2)F)cn2c(F)cccc2n1 C(C(=O)N1CCCC(N2CCN(C(=O)CC3CN(C)C3)CC2)C1)(C(C)C)SC c1(OCC(=O)N(C)CC2N(C(C(F)OC)=O)CCC2)ccc(C(C)C)cc1 N(C(=NCC(O)c1cccc(Cl)c1)NC1CC1)C1CC(OC(C)(C)C)C1 CSC1=C(C(=O)N2CCCCC2CNC(C2CC2(C)C)=O)CCCC1 C(=O)(C1=C(Cl)CCC(C)C1)N1C2(CNC(C3(COC)CC3)=O)CCCC(C1)C2 C#Cc1c[nH]nc1C(=O)NCC(CC1CCCC1)C(=O)NCC(C)CCO c1(C(N2C(C)CC(CNC(C(C)=C(C)C)=O)C2)=O)ccc(CO)cc1F C(CC(F)F)(C(=O)NCCc1csnn1)NC(=O)CC1CCCC1 CC1(C)CCC(CCNC(C2(NC(C3CN4CCC3C4)=O)CC2(C)C)=O)C1 C1(C(N2C(C(N(C)Cc3onc(CC)n3)=O)C3CC3C2)=O)C2CCCCCC12 N1(C(c2cc(CC)nn2C)=O)CCCN(C(C2(C)COCCO2)=O)CCC1 S(=O)(=O)(c1c[nH]c2cc(Br)cnc12)N1C(c2occ(C(C)(C)C)n2)CCC1 c1(C(=O)NCC(C)(C2CC2)NC(c2ccc(CC)o2)=O)ccc2c(c1)CCCC2 CCC(C(=O)NCCC(O)CNC(=O)CC1(N(C)C)CCCC1)C(C)C C1(CC(=O)NC(CC#C)(C)C)CCCCN1C(=O)CCC1CC1 c1(C(=O)NCCOCCCNC(CC=C)=O)cnncc1C(F)(F)F.C1CC1 C1(NC(=O)C(O)c2ccsc2)CCN(C(c2cnc(-c3ccoc3)s2)=O)CC1F C1(C(=O)NCC(C(C)O)O)CCC2CCC1N2C(c1ccc(O)cc1F)=O c1(CNC(CCC=CC)=O)cccc2c1CN(C(=O)CN1CCOCC1)C2 C(=O)(N=c1cc(Br)[nH][nH]1)c1cccc(Nc2nccc(C)n2)c1 C1(C(=O)NCC(=O)NCC(C)(C)n2cccn2)CC1[N+](=O)[O-] c1(CC)nc[nH]c1C(=O)NC1CCC1NC(=O)CCSc1nccn1C C1(C(=O)NCC(CNC(C2CN(C(C)C)C(=O)CC2)=O)O)CC12CCOC(C)C2 N1(C(c2nccc(CC)c2)=O)CC(NC(=O)CCC(F)F)CC12CCC2 c1(C(=O)NCC(CCOC)NC(c2c(CC)cno2)=O)c(Cl)cccc1Cl N1(C(CCCC(=O)NC)=O)CCC2C1CCCN2C(=O)C(C(C)(C)C)SC c1(NC(=O)NCCN(C(C)C)C(=O)OC(C)(C)C)ccc(Cl)c2occc12 C(=O)(NNS(=O)(=O)c1cc(Cl)ccc1Cl)N(C)CCc1ccccc1 c1(CC(N2CC3C(NC(C4CCCC4(F)F)=O)C(C3)C2)=O)cccc([N+](=O)[O-])c1 c1(C(=O)NCCCOCCNC(C(CC=C)C)=O)cnc2c(c1)COC2 c1(C(=O)NCCC(C(C)C)NC(C2(CO)CC2(F)F)=O)cc(F)c(F)cc1F C(c1ccc(OCC(F)(F)F)c(OC)c1)=CC(=O)NC1CC1C.N1(CC)CC1 CCCC(C#N)C(=O)NCCC1(O)CN(C(c2cnn(C)c2C(=O)OC)=O)C1 C1(C(C)=O)CCC(C(=O)NCC2CCN2C(=O)CC(=O)OCCC(C)C)CC1 N1(C(C(CC#C)C)=O)CCC(F)(F)C(CNC(=O)CC(=O)NCC(F)(F)F)C1 c1(C(N2CCC(CC)C2CNC(=O)CCCNC(N)=O)=O)[nH]ccc(=O)c1C C1(CC)(CC)CC(NC(=O)CCc2cnc(C)o2)CN1C(c1ccc(Cl)o1)=O CC1COc2ccccc2C1C(=O)NCC1CCN1C(C12CCC(CC1)OC2)=O N1(C(CCCC#N)=O)CCN(C(=O)CC23CNC(=O)C(C2)C3)CC1CCO c1(N2CCc3c(nc(C)o3)C2)nc(=NC2CSC(C)C2)[nH]c2c(C)nn(C)c12 c1(OC)cc(OC)cc(C(=O)NC2CN(C(c3ccn(C)n3)=O)CC2F)c1 CC1=C(C(=O)NCCC2CC(NC(C3CCCC(=O)N3)=O)C2)CCCC1 c1(CN(CC(C)O)CC)cc(Br)c(C)c(Br)c1 N1(C(C2(C)CCC(=O)C2)=O)CC2(CCC(CNC(C3(CF)CCOCC3)=O)O2)C1 N(C1CCCn2nccc21)C(=O)NC(c1ccc(Cl)cc1Cl)C c1(CC)cccc(NC(C2(N(C(=O)C=CCC3CCC3)C)CC2)=O)c1O C(CC(=O)N1CCC(N2CC(O)C2)C1)(C(F)F)NC(C(Cn1cncn1)OC)=O C=C=CCC(=O)NCC1COC(CNC(=O)CN2CCOCC2)C1 CC(C)C(CNC(=O)COC1CCCCC1)NC(c1ocnc1C1CCC1)=O N(C)(S(=O)(=O)N(C)C)CC(=O)N(CCOCCNC(C=Cc1scc(C)n1)=O)C N1(C(c2cnc(O)cc2O)=O)CCC2CN(C(=O)C(F)(F)C3CCCC3)CC12 Cc1nnc(OC(F)F)c(C(C)NC(=O)Oc2cccc(Cl)c2OC(F)F)c1C N1(C(C(C=C)(C)O)=O)CCN(C(c2n[nH]c(C)n2)=O)C(c2cc(F)ccc2F)C1 C1(C2(NC(c3nc(CC)sc3)=O)CC2)CCCCN1C(=O)C=C(C)Cl C1(NC(=O)CN2CC3CC3C2)CC12CCN(C(=O)CC1COCCO1)CC2 CCC(C)CCC(O)CC(=O)N(C)CCN(C(=O)CN(C)C(=O)C1CC1)C c1(OC)ccc(C(CC(N)=O)NC(=O)NC(c2cccnc2)C(C)C)cn1 C1(CNC(C2ON=C(C)C2)=O)(CNC(c2ccc(C3CC3)cn2)=O)CC12CCC2 N1(C(C(=O)NC)c2ncco2)CCC=C(c2cn(C(=O)OC)nn2)CC1 CN1CC(C(=O)N(CCCCNC(c2ccc(C(F)F)o2)=O)C)C(C(F)(F)F)C1 C1(CCC)(NC(C2OCCN(C)C2=O)=O)CCCN(C(=O)CC2CC3(CC3)C2)C1 c1(C(=O)NCC2C(C)(C)N(C(=O)CC3(C)CC3(Cl)Cl)CC2)cc2ncccn2n1 Cc1cc(N(C2C3CCC2CNC3)C(c2cncnc2)=O)c(C)cc1F c1(CC(=O)NC(CCNC(c2c(C(=O)OC)cn(C)n2)=O)C)cc(C)nc(O)c1 N1(C(C(C)NC(C)=O)=O)CCC2(CCN(C(C3CCC(C)(C)O3)=O)CC2)C(C)C1 C1(C(=O)NCC(C)(C)NC(C(C)CSc2ccc(F)cc2)=O)CC2CCC(C1)S2 CCC1=NOC(C(=O)NCC2CCN2C(c2cc(C)nn2-c2ccccc2)=O)C1 C1(OCC)CC(NC(N2CCn3nccc3C2)=O)C12CCCC2 N1(C(c2ccc(CC)[nH]2)=O)CCC(NC(C2CC(=C3CCC3)C2)=O)C(CO)CC1 c1(OCC)ncc(F)c(=NC(=O)C2CC3(CC3)CN2C(c2ccc(Cl)cn2)=O)[nH]1 c1(C(N2CCC(C(=O)NC(CC#C)CC(F)F)C2(C)C)=O)cnc(C)c(C#N)c1 N1(C(C(=O)NCC)=O)CCCN(C(c2ccc(C)c(C(F)(F)F)c2)=O)CC1.NC c1(OC)cncc(C(=O)NC2CCC(NC(c3c(Br)cnn3C)=O)C2)c1C Cc1ncc2n1CC(C(=O)NCC=CCNC(=O)CC1CSCCS1)CC2 C1(CN(C2CCCC2)C(COC)=O)CN(C(=O)C=CC(C)(C)SC)CC1C CN1CCCC(O)(CC(=O)NCC2CN(C(c3cn(CCF)nn3)=O)CCO2)C1 C(N=c1[nH]cnc2c1CCC2)C1(CNC(C(CC)OCC)=O)CCC1 C1(NC(CC(=C)I)=O)CCSC12CN(C(c1ccon1)=O)C2 Cn1c(C(=O)NCC(C2CCC2)NC(=O)C(F)=CC2CC2)cc2cc(Cl)ccc12 C(=O)(C(O)C(C)(C)C)NC1(Cn2nnc(C)n2)CNC(=O)C1.n12cc(nn1)CC2 C(=O)(C(=O)C(F)(F)F)NC1CN(C(C=Cc2ncn(C)c2)=O)C1 C1(C(N2CCC(CCNC(=O)CSC(F)(F)F)C2)=O)CC2CCC(C1)O2 C1(NC(c2cc[nH]n2)=O)CCC2(CCN(C(=O)Cn3cnccc3=O)C2)C1 C1(C(=O)NCC(C(C)C)NC(c2cncc(F)n2)=O)CCCC(F)(F)C1 CC1CN(C(c2coc(Br)c2)=O)CCN1C(c1coc(CC2CC2)n1)=O C1(C(N(C2CCCN(C(=O)C(C)(C)C3CC3)C2)CC)=O)CCc2ncccc2C1 c1(OC)ccc(S(=O)(=O)NCCCc2nc(C(C)C)n[nH]2)c(F)c1F N1(C(C(=O)NCC(C)C)=O)CCC2(CC1)CN(C(=O)C(C)CS(C)(=O)=O)CCC2O Cc1ccnc(CN(C)C(C2CCN2C(c2cnsc2)=O)=O)c1 CC1=NS(=O)(=O)NC=C1C(=O)NC1(C)CCN(c2ncc3ncnc-3[nH]2)C1 C1(C(NOC(CC)C)=O)C=CCN(C(=O)Cc2cncnc2O)C1 C(CCC(C)CO)N(C(c1ccc(COC)o1)C(=O)NCCC(=O)OC(C)C)C N1(C(c2c(OC)nn(C)c2)=O)CCC2C(CCCN2C(c2nnsc2C)=O)C1 C1(NC(C2CCCN(C)C2)=O)CCN(C(c2cccc(C3CC3)c2)=O)C12CC2 C1(C(=O)NCCC(C)N(C)C)(NC(=O)CCc2nccn2C)CC(F)C1 C(CCCCC(=O)NCCC(=O)NC(C)C)NC(C(C)OCC#C)=O C(CN(C)C)(C(=O)N1CC(N2CCC2)C1)NC(C(c1ccnn1C)C)=O CC1CN(C(=O)COc2cccc(Cl)c2Cl)CCC1CNC(c1cnsn1)=O c1(C(N2CCC(C(=O)NC(CC=C)CO)C(O)C2)=O)cc(Cl)cc([N+](=O)[O-])c1C C(C)(CCC(c1nnnn1C1(C)CC1)NCc1nncs1)OC C(=O)(CCC(=O)NC1CCCC1NC(=O)Cc1nnc(C)o1)OC c1(C(=O)NCC2(NC(C3C(C=C(C)C)C3(C)C)=O)CC2)nnn2c1CSCC2 N1(C(C(CCC)O)=O)CC2(CCCC2)C1C(N1CCN(C)C(CC)C1)=O n1(C(C)OCC)nc(Br)c(CNC2(O)CCN(c3ccccc3)C2)c1Br C1(C(N(CCCCCNC(c2nnc(Cl)cc2N)=O)C)=O)CN2CCC1(C)CC2 N1(C(c2cc(C)on2)=O)CCCC2CCN(C(c3cn(C(C)C)cc3C)=O)CC12 N1(C(C2N(C(C)C)CCC2)=O)CC2CN(Cc3c(F)cccc3C#N)CC2C1 N1(C(c2ccc(CC)nc2)=O)CCC(NC(c2ccccc2C)=O)C(F)C1 C1(CC(=O)N(C)Cc2cnn(C)c2)CCC(=O)N(C(C)(C)C)CC1 N1(OCC)CCCC(C(=O)NCCC2CC(NC(=O)C(CC)N(C)C)C2)C1 C12(C(=O)NCC3(CN(C)C(C4CCCC4C4CC4)=O)CC3)CC=CCN1CCC2 O=C(C#CC1CCOC1)N1CCC(CCC2CCCN(C(=O)C3CC3)C2)CC1 CCCCC(O)C(=O)NCCCC(CCC)NC(=O)Cc1cc(C(C)C)no1 N1(C(C(C=CCCC)O)=O)CCC2(CCN(C(c3nc(Cl)ccc3N)=O)C2)C1 C12(CNC(C=CC(CC)C)=O)CCCC1N(C(=O)COC1CCCC1)CC2 Cc1cc(C(=O)NC2CCC2NC(=O)CCCC2CCOCC2)nn1C(F)F n1(CCNC2(CCO)CCC(C)C2)c(O)nc2ccccc12 C1(C(=O)NCC2(CC)CCCCO2)CC(C)CN(C(=O)C(N)=O)C1 C1(C2CCCCC2)(C(=O)NCC(CC)NC(=O)Cc2cncn2C2CC2)CC1 N1(C(CC2(C=C)CC2)=O)CC2=C(C1)CN(C(c1cc(C)c(C)o1)=O)C2 C(=O)(C(CC)C(=O)OC)N1C(NC(c2nc(OCC)oc2)=O)CC(OC)C1 C(=O)(C1=CCCOCC1)NC(C(C)C)CC(=O)NCC1Cc2nccn2C1 O=S(=O)(c1ccc(NCc2ccc3c(c2)CCCC3)c(F)c1)Nc1ccns1 Cc1c(C(=O)NCC23CCC(CN2C(c2ccnnc2)=O)C3)[nH]c2ccccc12 CC(C)CCCOCC(N1CCCC1C(=O)NCC(C)(C)C1CCCC1)=O Cc1cc(C(=O)NC2CCCC2NC(c2cc(C(N)=O)[nH]n2)=O)c(C)[nH]1 Cc1nc(Nc2cnn(C3CCCCO3)c2)ncc1Br C1(NC(=O)CC2CCC(=O)N2)C=CCN(C(c2nsnc2O)=O)C1 c1(CC)c(C(=O)NCC2CC(C)N(C(=O)C=NOC)C2)cnn1CC c1(C(N2CCCC(CCNC(C3=CC(C)CC3)=O)C2)=O)onc2c1CCCC2 N1(C(CCCCC(N)=O)=O)CC(CNC(=O)CSC(F)(F)F)C2CCCCC12 c1(C(N2CC(O)(CN(C(C(C)C#N)=O)C)C2)=O)nccc(Cl)c1F C12(C(=O)NC3C(NC(C=C(CC)CC)=O)CCCC3)CC3CC1C2C3O C1(CNC(C(=O)NCCOC)=O)C(C)CCCN1C(=O)CCC(F)F C1(C(N(CCCO)C)=O)CC(N=[N+]=[N-])CN1C(C12CCCC1C2(F)F)=O C1(CNC(CC(C)c2cccnc2)=O)CCCCN(C(=O)Cc2cnccn2)C1 n1(CC)nnc(C)c1C(=O)NCCCC1CN(C(=O)Cc2n[nH]c(=N)s2)CCO1 C1(OCC)CC2CN(C(C3CC4CC4N3C(=O)CC3CC(N(C)C)C3)=O)CC12 C1(NC(Cc2c(C)cco2)=O)CCN(C(=O)C=C2CCN(C)CC2)CC1C(C)C C12(NC(=O)Cc3cscn3)CCCC1(F)CN(C(C1CC1C(N)=O)=O)C2 C(=O)(C(CNC(=O)CCC=C(C)C)CC(C)C)NCC(C#C)(C)C CCS(=O)(=O)C=CC(=O)NC1COCCN(C(=O)CC2CC3CCC2O3)C1 c1(C(=O)NC(C2(O)CCN(C(=O)Cc3cc[nH]c(=N)c3)C2)C)ccncc1F c1(C(=O)NC2C3CN(C(c4cncn(C)c4=O)=O)CC32)c[nH]c2cccc(Cl)c12 S(=O)(=O)(c1ccccc1C(=O)O)N1CCC(C(=O)Nc2cccc(CC)c2O)C1 c1(-c2c(C(=O)OC)cncc2)cnn2ccc(C)cc12 C1(CNC(C(C)=C2CCC2)=O)N(C(=O)CC2CC(C)(C)CO2)CCCC1(C)C c1(C(N(CCCNC(=O)C(c2ccccc2F)C)C(C)C)=O)ncc(F)cc1N c1(C(N(C)C(C2CC2)C2CC2)=O)c(CNC(=O)C(F)C2CCOC2)nnn1C C1(C(=O)NCCCOC)CC2(C1)CN(Cc1ccc(C)cc1)C2 N1(C(CCNC(C)=O)=O)CC2CCC(C1)C2NC(c1cccc(Br)n1)=O CC(CC(=O)NCC(O)CNC(c1ccc(=N)[nH]n1)=O)C(F)(F)F N1(C(c2c(OC)ccc(Cl)c2)C(=O)NC2CCC2)CCc2ncn(C)c2C1 c1(C(=O)NC2C=CCN(C(C=C(CCC)CCC)=O)C2)cnc2ncccc2c1 CC1CN(C(=O)C(C)c2ccsc2)CCN1C(=O)Cc1csc(-c2ccoc2)n1 c1(C(=O)NC2C(CC)N(C(C3CCC4CC34)=O)CCC2)ccn2ccnc2c1 C1(C(N2CC(CO)C(CO)C2)=O)CCN(C(=O)CC2CCCCC2O)C12CC2 N1(C(COCCCCC)=O)CCC(C)(C)C(NC(=O)CC(C)n2ccnc2)C1 C(=O)(CCC(F)(F)C(F)F)NC(C)(C)CCNC(=O)C1=CCCCC1 C1(CN(C)C(C2(C)CC=CCC2)=O)CCCN(C(c2ccsc2C#N)=O)C1 C1(C(=O)NCC2CCCCO2)CCC2(CC2)N1C(c1cc(F)c[nH]1)=O C1(C(N2CC(CNC(C3CC4CCC3CC4)=O)C(O)C2)=O)CC12CCOCC2 c1(OC)ccc(F)c(C(=O)NC2CN(C(c3cnn(CCO)c3C)=O)C3CC23)c1 S(=O)(=O)(c1ccc(NCC2CC(n3ccnn3)C2)c(Br)c1)NCCC(CCC)C C(CC(C)(C)C(=O)N(CCC(=O)N(C)C(c1ccccc1)C)C)OC C(CN(C(=O)CCn1cc(CCCOC(=N)O)nn1)C)(C(C)C)OCC C1(CNC(=O)CCc2ccncc2)COCCN1C(C1CC1C1CCC1)=O C1(C(=O)OC)CN(C(C(=O)NC2CC(F)(F)C2)C2CC2Cl)CC1C1CCOCC1 N1(C(C(CC=C)(C)C)=O)CC(CNC(C2C(CN=[N+]=[N-])C2(C)C)=O)CC(C)(C)C1 N1(C(c2c(CC)ncnc2)=O)CC(CNC(=O)C(C)C(C)C)C2(CC2)C1 c1(C(=O)NCC23CC(NC(c4ncn(C)n4)=O)(C2)C3)sc2sccc2c1Cl N1(C(c2c(OC)nccc2)=O)CCCC(F)(C(=O)NC2CCCCCC2OC)C1 Cc1cccc(CC(N2CCOC(CNC(=O)COC3CCCCCC3)C2)=O)c1 c1(N2CC3CC(NC(c4c(C)cc(SC)o4)=O)C3C2)nc2ccc(C)nc2s1 C(=O)(CCCC(C)(C)NC(=O)CC1CCCCO1)NCc1cc(OC)no1 C#Cc1ccc(Cl)c(C(=O)NCCC2CN(C(=O)C(F)OC)CCS2(=O)=O)c1 CC(F)(F)CCCCN=C(NCC1(S(C)(=O)=O)CC1)NC(C1CC1)C1CC1 Cc1cc(C(=O)NCC(C2(O)CN(C(=O)Cc3csc(Cl)n3)C2)(C)C)sn1 N1(C(c2c(OCC)ccs2)=O)CCN(C(=O)Cc2ccc(Br)cn2)CC1 N1(C(C(C2CCOC2)OCC)=O)CC2(C1)CN(C(=O)C(C)(COC)COC)C2 c1(SC)ccnc(N2CC3CC3(CNC(C3CCCN3Cc3cccs3)=O)C2)n1 c1(C(=O)NCC(CCOC)NC(CCCC=C)=O)oc2ccccc2c1COC CC1CCN(C(=O)CC2C3CN(C(=O)C4=CCCC4C)CC23)C1(C)C c1(C(N(C)C)=O)ccc(C(=O)NC(c2nncn2C)(C)C)c(O)c1 C[Si](C)(C)C#Cc1cccc(NC(C2CC2NCc2cc(Br)ccn2)=O)c1 C1(C(=O)NCCCC(C)(C)NC(CC(=O)OC(C)(C)C)=O)CCc2nnnn2C1 N1(C(c2c(CC)con2)=O)CCC(CO)(CNC(C2CCOC2C(C)C)=O)CC1 C1(O)(CN(C(=O)CNC(=O)C2CC2)C)CCN(C(C2CC=CCO2)=O)C1 C(CCCCOC)(c1n(CCCCCC)nnn1)NCC1CCCN1S(C)(=O)=O C(=O)(CCC(=O)N(CC(C)NC(C1OCCC1C(F)(F)F)=O)C)OCC c1(C(CCC#N)C2CCC2)ccc(Cl)cc1.N1(C(CC)=O)CC(C=O)(C)C1 N1(C(c2cc(C)nn2C(F)F)=O)CCC(NC(c2scc(C)c2Cl)=O)C(F)C1 C1(C)(C(=O)NC(C2CCN(C(=O)Cn3cnnn3)C2)C)CC2CCC(C1)S2 O=C(C1=CC2CC(C1)CC2O)NC1CCN(C(=O)CCN2CCCCC2)CC1F c1(C(N2CCC(OCCNC(CS(=O)(=O)NC)=O)C2)=O)cnc(N)c([N+](=O)[O-])c1 CC1(C)CC=C(C(=O)N2CC(C(=O)NC3CCC34CCCC4)C3(CCC3)C2)CC1 c1(CCC(N2CCC(C(C)(C)NC(=O)C(C)SC(F)(F)F)C2)=O)ccccc1F N1(C(c2c(C)nc(-c3ccccc3)o2)=O)CC2CCC1CN2C(=O)C(F)CC(C)C C1(NC(CCCCC=C)=O)CCN(C(C2(S(C)(=O)=O)CCC2)=O)CC(O)C1 C1(NC(C2(O)CC(C)(C)C2)=O)CN(C(=O)CSCC2CCCO2)C(C)(C)C1 [N-]=[N+]=NCCCC(=O)NC1COCC1NC(=O)CCc1ccc(F)cc1Cl C(c1ccccc1F)=CCC(=O)NC(CNC(C(C)CN1CCCCC1)=O)(C)C C12(NC(CCS(C)=O)=O)CCC1CN(C(=O)CCCC1CCCC1)C2 Cc1nn(C)c2c(N3CCC(CC(F)F)C3)nc(N3CCC(=O)N(C)CC3)nc12 C(=O)(CCC(F)(F)CN=[N+]=[N-])NCC1CCN(C(c2cnc(C)o2)=O)C1 CC1CCC(=CC(=O)NC2(CF)CCN(C(C3(n4ccnn4)CC3)=O)C2)CC1 C(=O)(CCCCC#N)NCCC(C)(C)NC(C12CC(C)(C1)C2)=O c1(N(CCOCCOC)C)cccc(CNC2(C(=O)O)CCCOC2)c1 c1(NC(C(=O)N(c2ccc(CC)cc2)CC)=O)cc(C)cc2ccc(CC)cc12 CCS(=O)(=O)NCCNC(=O)C(C)NC(=O)COC1CC(SC)C1 CC1=CC(C)C(c2c[nH]nn2)CC1.C(CCC(C)(C)C)C1CCNCC1 C(=O)(CC(CC(=O)NC(=O)C(C)(F)F)SC)NCC(CCN(C)C)OC C1(NC(C(C)O)=O)CCN(C(c2cc(F)ccc2N2CCC(O)CC2)=O)C1(C)C Cc1ccc(C(=O)NC(C)C(CO)NC(=O)C(O)C(F)(F)F)c(C2CC2)c1 c1(C(N2CC(CNC(C=CC=CC)=O)(OC)C2)=O)ccccc1N1CCCC1 c1(C(C(=O)NCC2N(C(CCC(C)N(C)C)=O)CC2)=O)cc(F)c(F)cc1F C1(C(=O)NC(C(=O)NCCC)CC)C2CCN(C(=O)C(CSC)OC)CC12 C1(NC(C(C)C2CCC2)=O)CCC(C)(NC(=O)Cc2ccncn2)CC1 C1(C(N2CCC(CNC(c3cnco3)=O)C23CC3)=O)CC2CCCCCCC12 Cc1nccc(C(=O)NCCCN(C(=O)C(C#N)C(C)C)C2CC2)c1C Cc1nc(NC(N2CCC(CN(C(=O)COCC3CCCO3)C)C2)=O)n(C)n1 C1(C=O)CC2CCC1N(C(=O)C#CC1CCOC1)C2.c1(CSCC=O)ccncc1 N1(CC)CCCC1C(=O)NCCOC1CCN(C(c2cc(Cl)n[nH]2)=O)C1 c1(CC(N2CCN(C(c3sccc3F)=O)C(C)C2)C)ccc(Br)cc1F C1(C(=O)O)CC2(CCC2)CN1C(c1ccc(C(F)(F)Cl)cc1)=O N(C(=NCCc1cccnc1)NCC1CC1)C(c1ncccc1F)C Cc1c[nH]c(C(N2CC(C(C)(C)O)(CNC(C3CCN3S(C)(=O)=O)=O)C2)=O)c1 C#CC(CNC(c1cc(CCNC(=O)CCC2CCC2)on1)=O)CC1CC1 N1(C(c2ccc(CNC(C(C)(C)C(F)F)=O)cc2)=O)CCC(C2CCOC2)C1 N1(C(c2nnc(C)s2)C(=O)NCCC#N)CCOC(CN(C)C)C1 N1(C(c2c(CC)nccc2)=O)CCC(NC(=O)CNc2nnco2)C(O)C1 N1(C(c2n(C(CC)C)ncc2)=O)CC(NC(=O)Cc2cncs2)CCC1C C12=CC=C(C=C1)C2.N1(N(C)C(=O)NCc2c(C)noc2)CCC(C)CC1 c1(CCC(N2C(C(CCC)=O)CCC2)=O)ccc(C)c(OCC)c1 N1(C(C=CC=CCC)=O)CCOC(C(N2CCN(CC(C)O)CC2)=O)C1 Cc1cccc(C2C(C)CN2c2nc(C3CCC3)cs2)c1 n1(CC(N2CC(CNC(CCCSC)=O)C(C(F)(F)F)C2)=O)ccc([N+](=O)[O-])n1 Cn1ncc(=NC(=O)C2(O)CN(Cc3c(Cl)cnc(Cl)c3Cl)C2)[nH]1 C=CCCCCN(C)C(C1CC1C(C)NC(=O)C(CC1CCCC1)OC)=O CCC(CC(=O)N1CCCCC1CC(=O)NOCC(C)(C)O)OC CC1CC(C)(C(N2CCC3(CC3)CC2C(=O)O)=O)CC(C)O1 N1(C(c2cccc(N)n2)=O)CC2CCCC(C1)N2C(c1nocc1Cl)=O C12(NC(C3ON=C(C)C3)=O)CCCC1N(C(c1cccc(C(C)(C)C)c1)=O)CC2 N1(C(c2cnc(OCC)nc2)=O)CCC(C2CCN(C(=O)C=CCOC)C2)C1 c1(C(N2CC(NC(c3cncc(-n4cccc4)c3)=O)C2)=O)cc2n(c1)CCCC2 N1(C(C(COC)N(C)C)=O)CCC(C(=O)NCC2(F)CC(CO)C2)C12CCC2 c1(C(=O)NCC2N(C(C3CC(OC)C3)=O)CC(C)CC2)nc(C)c(C)[nH]c1=O c1(C(=O)NC2CCN(C(C3=C(C)OCC3)=O)C2C)ccc2scc(C)c2c1 N1(C(=O)CC2(C)CCCCC2)CCCC(O)CC1.CC1C=CC(=O)N1 n1(CCC)ccc(=NC(=O)CC(C(F)F)NC(C2(C(=O)NC)CCC2)=O)[nH]1 C(=O)(CC(C)(C)CCOC)NC1(CCNC(CC2ON=C(CC)C2)=O)CC1 c1(CCCC)ccc(C(N2CCCC(C(=O)NC3(CNCC=[SH]C)CC3)C2)=O)cc1 O=C(CC1CCN(C(c2cnco2)=O)C1)N=c1cc(C(F)(F)F)[nH][nH]1 c1(C(=O)NC2C(NC(c3ccc(OC4CC4)cc3)=O)CC2)ccccc1F C1(F)(NC(C(C)OCC2CCCO2)=O)CC(NC(=O)CSc2ccncc2)C1 N1(C(CC(CC)(F)F)=O)CCC(F)(F)C(CNC(=O)C(C(C)(C)C)N(C)C)C1 C#CCC(C)(C(=O)N1CCC(C)(N(C)C)CC1)NC(c1ccc(C)o1)=O C#CCC(CC(F)F)NC(=O)C(C)CN(C)C(C1CCCN1C=O)=O C(CN=c1[nH]c(Cl)ncc1[N+](=O)[O-])(C(C)(C)C)NC(c1n(C)nc(C(F)F)c1)=O N1(C(C(C)(C2CC2)OC)=O)CC(CNC(=O)CCCn2ccnc2)CC(C)(C)C1 c1(C(=O)NCCNC(C2CN(CSc3cccnc3)CCN2)=O)ccc(Cl)nc1 C1(CC=C)(NC(C2CCC2)=O)CCN(C(=O)CCC)C1 c1(C(=O)NCC2N(C(CC(CC)C)=O)CC(O)C2O)nc[nH]c2ncnc1-2 C1(C#CC(=O)NC2(CNC(=O)CC3C=CCC3)CCCC2)(CC)COC1 C1(C)(CNC(C2C(C)(C)C2(F)F)=O)CCCN(C(=O)CCS(N)(=O)=O)C1 CC(C)C(O)CC(=O)NCC(C)(C)CCNC(=O)C(C)(C)C(C)O N1(C(c2c(C)[nH]cc2)=O)CCN(CCCNC(C2(OC(C)C)CCOC2)=O)CC1 c1(OC)c(Cl)nc[nH]c1=NCC1C2CN(C(C3CSC3)=O)CC12 C1(CC)C(C(=O)N(C)CCOC(F)F)CCN1C(c1oc(C)cc1C)=O CCCCC(C(=O)NCc1cccs1)NC(=O)C(CC)NC(C)=O C(=O)(C1=CCCC1C)NC1C(NC(c2c(C)nc(-c3ccsc3)s2)=O)CCCC1 C1(C(C(=O)NC(C(=O)NCCC(C)N2CCC2)C2CCCC2)=O)CCCCC1 C(=O)(CCCCc1cn(C2CCOC2)nn1)NCC(C(=O)O)Nc1cn(C)nc1 CC(C)(CNC(c1sc(CC2CC2(F)F)nc1-c1ccccc1)=O)C(=O)O C(CC(O)CNC(c1cc(Br)no1)=O)NC(C(C)OCC)=O c1(C(=O)NCCCCNC(C(C)C2CCCO2)=O)cccc(OCCOC)c1 c1(C(N2CC(NC(CC(C(=O)OC)(C)C)=O)C(C)C2)=O)cc2cccc(C)c2o1 C1(C(=O)NC(C)CCNC(=O)CC2(C#N)CCC2)(OC)CCCC1 N1(CC(=O)Nc2ccc(OC3CCCCC3)cc2)CCOC2(CC(O)C2)C1 N1(C(C(n2c(C)ncc2)C)=O)CC(NC(=O)CN2CC=CC2)CCC(O)C1 c1(CC(=O)NC(CC)CNC(c2c[nH]nc2OC)=O)c(C)nn(CC(C)C)c1C Cc1n[nH]c(C)c1CCC(=O)NC1CC1NC(=O)CCn1ncn(C)c1=O C1(CNC(Cc2cc(CC)no2)=O)CC(CO)N(C(=O)C=Cc2nccs2)C1 n1(CCCC)nnnc1C(CC1CCCC1)NC(c1sccc1Cl)C C(=O)(C1=CCC(C)CC1)NCCC(C)NC(C(c1nccc(C)c1)(F)F)=O CCCC(CCCNC(c1cc(C)nc(C)n1)=O)Nc1ncnc(Cl)c1C(C)C C1(NC(CCOCCCC(CO)N(C(=O)C(=O)NC2CC2)C)=O)CCCCC1 Cc1ccc2c(c1)CC(C(=O)NC(C)CNC(c1sccc1Br)=O)S2 C1(OC)CN(C(C2CC2CC(C)C)=O)CCC1NC(c1cccc(Cl)c1F)=O N1(C(C(CC)COC)=O)CCC(CNC(=O)C(C)(F)c2ccon2)C1(C)C c1(CCC(=O)NC2C(NC(CCC(CC)CC)=O)C2)c(C)nc2ccnn2c1C c1(C(N(CC(C)N(C(=O)C(C)n2ccnn2)C)C)=O)nccnc1N C(=O)(CC(C)C(=O)NCC1CCN(C(c2ccc([N+](=O)[O-])o2)=O)CC1)OC CCC(CCOC)C(=O)NC(C1CC(NC(C2(C(C)(F)F)CC2)=O)C1)C c1(SC)nc(N2CC(F)CC2CNC(c2ccnc(OC(F)F)c2)=O)ncc1C CCCC(C)C(=O)NCCC1CSCCN1C(=O)Cc1conc1C c1(C(N(C2(C(=O)NC3C(C)CC3)CCSC2)C)=O)sccc1C#N C1(C(=O)NC(c2ccsc2)C)CCN(C(C2(CC3CCC3)CC2)=O)CCO1 c1(C(C(=O)NC(C)(C)C)N(C(C(=O)OC)C)C)occc1Br C1(NC(C(C)(C)OC)=O)CCN(C(=O)C(F)C(F)(F)F)CCC1c1ccccc1 c1(C(N(CCCNC(CC2CC(=O)C2)=O)C2CC2)=O)ccc(OC(F)F)cc1 c1(N2CCC(C)(C(=O)NC)CC2)nc2cccc(F)c2c(=NCCCF)[nH]1 C1(C(C)O)CCN(C(=O)C(F)CC2CN(C(C3CCN3C)=O)C2)CC1 c1(C(=O)NC(CCNC(COCCOC)=O)C)cc2c(cc1Cl)OCCO2 N1(C(C(C)=O)=O)CC2CC(C1)N(C(=O)Cc1ccc3nn[nH]c3c1)C2 n1(CCC(=O)NC2CCCC(NC(c3cccs3)=O)C2)cnc2ccccc12 N1(CC(C23C(C)(C)C(CC2)CC3)=O)CCN2CCNCC2C1 CC1CCN(C(=O)CNC(=O)C2CC2)C1CNC(=O)C(=O)NCC1CCC1 c1(N2CCC(C)C2)ccc(S(=O)(=O)N2CCc3ccccc3C2)cc1Br c1(C(N2CCC(C)(NC(C3C=C(C)CS3)=O)CC2)=O)ccc(C#N)cc1F C(=O)(C(C)CC(F)(F)F)N1CC(CC)N(C(C2CCN(C(C)=O)CC2)=O)CC1 N1(C(C)=O)CSCC1C(=O)NC(C)(C)C(C)NC(=O)Cc1ccc(Cl)s1 CCC(CC(=O)NCC1CC(NC(=O)CC2CCS(=O)(=O)C2)C1)C(C)C N1(C(c2ccc(Cl)s2)=O)CC2CCCC2(C(=O)NC2C3COCC23)C1 CC(C)(C)CC(O)CNC(=O)CC(CNC(=O)C1=CCOCC1)C1CCC1 N1(C(CCCC)=O)CCCC(C)(NC(=O)C(C)Oc2ccc(F)nc2)C1 N1(C(c2c(C(C)(C)C)con2)=O)CC2CC(c3ccccc3)C(C2)C1 C1(C(=O)NCC2CC(NC(C(CSC)OC)=O)C(O)C2)CC(=O)N(C)C(=O)N1 c1(C(N2CCC(CC=C)(NC(C3CCCO3)=O)C2)=O)sc2ncccc2c1N Cc1c(C(N2CCC(C)C2CNC(C2(F)CC2)=O)=O)[nH]c2cc(Cl)ccc12 c1(NC(C(CC)(C)CNC(=O)CCc2cscn2)=O)cnc2ncnn2c1 CN(C(=NCCN1CCOC(C)(C)C1)NC1CCCSC1)Cc1ccnn1C C1(O)(C(C)NC(CC(CC)C)=O)CCN(C(C23CCC2CC3)=O)CC1 c1(C(N2C(CC(N3C(C(=O)O)CCC3C(F)F)=O)CC2)=O)ncnc(O)c1F N1(C(C(C)OCCCCCC)=O)CC2(CNC(=O)CSCCCC)CC(F)(C1)C2 N1(C(C(CC)N(C(=O)CC2CC2)C)=O)CCC(CCF)CC1 C1(C(=O)NC(C(C)C)CNC(c2cnccn2)=O)COc2ccc(Br)cc2C1 C1(NC(C=Cc2n(CC)ncc2)=O)CN(C(c2cc(C)ns2)=O)CC1(C)C c1(C(=O)NC2C(NC(=O)CN3CC=CC3)CCOC2)ccc2ccccc2n1 c1(CC(N2CC(O)(C(C)NC(Cc3c(C)non3)=O)C2)=O)cccc(F)c1Cl C(CN=c1[nH]c(C)cc(=NC2CCN(C)C(C)C2)[nH]1)=CCCOC c1(CNC(C(N2C(C)CCC(C)C2)=O)=O)ccc2c(c1)N(C)CCC2 C#Cc1ccc(C(=O)NC2CC=C(C(=O)NCC(c3ncc[nH]3)C)C2)cc1 c1(C(=O)NCCOCCC=C)ccc(NC(C2CCOC2COC)=O)cc1 C(CC(C)(C)C)(C(=O)N1CC(N2CCCC2=O)C1)NC(c1nn(C)c(C#N)c1)=O C1(O)(C(C)NC(c2ncccc2F)=O)CCCN(C(=O)CC2(O)CCOCC2)C1 N1(C(c2c(C)n[nH]c2)=O)CC(C(=O)NCC=C2CCSCC2)CC12CCC2 C(=O)(C1=CCCCC1P(C)(C)=O)NC1CC(O)(CNC(c2c(C)cn(C)c2)=O)C1 N1(CC)CCCN(C(C2(C)C=CCN2C(C2CS(=O)C2)=O)=O)CC1=O C1(C)(CC)CN(C(c2c[nH]nc2CCNC(C2COC(=O)C2)=O)=O)CCO1 c1(C(=O)OC)ccc(O)nc1N1CCCC1CCNC(c1cccnn1)=O c1(-c2cccc(N(C)C)c2)cnc(F)c(C(=O)Nc2ccnn2C(C)(C)C)c1 C(=O)(CCC(CF)CF)N1C(C(=O)NCCCCCC)CC(CC)CC1 C1(CNC(C(C)(C)c2cscn2)=O)CC2(CCN(C(=O)C(F)(F)CO)C2)CO1 CC1CCC(CC(=O)NCC2CCC(C(=O)NOCC(O)CO)C2)CC1 CC(C)C(C)CC(=O)NCCC1CC(NC(c2ccnc(F)c2O)=O)C1 n1(CCCC)nc(C(=O)NC2CC(C)(NC(=O)C#CC(C)(C)C)C2)ccc1=O C1(CNC(c2c(CC)occ2)=O)CN(C(C2CCCC23CC3)=O)CC1C(F)(F)F C1(C(N(C2CCN(C(=O)Cn3cccc3)CC2)CCC)=O)CC=C(C)CC1 N1(C(C=C(C)Cl)=O)CC(NC(=O)C(C)(F)F)CC12CCC2 c1(N(C)C)ccc([N+](=O)[O-])c(C(=O)OCc2nn[nH]n2)c1 c1(C(N2CCC(C(C)NC(c3c(CC)cccc3)=O)C2)=O)ccc2nnnn2c1 c1(NCc2c(C)ccc(C)n2)[nH]c(=NCCCCCCO)nc2c1ncn2C Cc1occc1C(N1C(C(=O)NCC2CSCCO2)CC1C)=O c1(C(=O)NCC(N(C(CCCSC)=O)C)C2CC2)cnc(SC)n1C CCCCC(C)C(=O)NCC(CNC(=O)C1=COCCC1)CO C1(OC)CC(CNC(=O)Cc2cnc[nH]2)N(C(=O)C=CC(=O)N(C)C)C1 N#Cc1ccc(C(N2CCC2CNC(=O)CCC2CCCC(O)C2)=O)[nH]1 CCC(C)CCCC(=O)NCC1(C)CN(C(c2ccc(F)c(OC)c2)=O)CCO1 c1(C(N2C(C(N3CCCC(OCC#C)C3)=O)COCC2)=O)ccnc(Br)c1Cl c1(CC)[nH]c(=N)sc1C(=O)N(C1CCCN(C(=O)C=CC(=O)N(C)C)C1)CCO C(=O)(CCC(F)(F)C(F)F)N1CCN(C(CN(C(CCC(=C)C)=O)C)=O)CC1 C1(CC(=O)NC(CC(C)NC(C2(OC)CCCC2)=O)C)CC2CCC1C2 c1(C(C)=O)cc([N+](=O)[O-])ccc1N1CC2CC(NC(C3C4COCC34)=O)CC1C2 N1(C(CC)=O)CCCC(C2CCCCN2C(=O)CC(=O)NCC)C1 N1(C(c2ccnc(OC)n2)=O)CCC(NC(=O)CSCCN(C)C)C12CCC2 N1(CCCCNC(=O)Nc2c(C)nc(C)s2)C(=O)C2C3C=CC(C3)C2C1=O c1(C(C)C(=O)NC2CC(NC(C3CCOC(=O)N3)=O)C2)cc2ccccc2o1 c1(C(=O)NCC(C2CCN(C(C3CC34CC4)=O)CC2)(C)C)cc2n(c1)CCSC2 c1(NC)c(C(=O)NC2CCCCN(C(=O)C3=CCCO3)C2)cccc1N c1(C(N2CC(NC(C3C(C=C)C3)=O)C(OC)C2)=O)cccc(SC)c1[N+](=O)[O-] N1(c2nnc(CCOC)s2)CCC2(CCCN(C(=O)C3=C(SC)CCCC3)C2)C1 C1(C(=O)NCC(C(C)C)NC(C2(CC3CC3)CC2)=O)(OC)CCCOC1 C1(NC(c2c(C)nco2)=O)CC(CNC(=O)CCCc2nncn2C)C1(C)C N1(Cc2ccc(C)o2)CCC2(CC2C(N2CCN(c3ccccc3)CC2)=O)C1 n1(C(C(=O)NC(C2N(C(CN(C)CC)=O)CCC2)C)C)c(=O)oc2ccccc12 C1(NC(C(CC)(C)F)=O)CCC2(CC1)CC(NC(c1cccc(NC)n1)=O)C2 c1(C(N2CCC(CC=C)(C(=O)NCCC3CCSC3)C2)=O)[nH]ccc(=O)c1C C1(C(=O)Nc2c(C(C)C)cncc2)CC(C)CN(C(c2cnc(F)c(Cl)c2)=O)C1 C1(N(C(CC=CC)=O)C)CN(C(=O)C(O)COC)CC1(C)C N1(C(c2cc(C(C)C)sn2)=O)CCN(C)C(CNC(=O)C(C)c2cccs2)C1 c1(NC)c(C(=O)NCC2C3CN(C(C4C=CCC4)=O)CC23)nnc2ccccc12 Cc1ncc(C(N2CC(CNC(=O)CNC(=O)NC3CC3)C(C)C2)=O)cc1N c1(C=O)nc(C)nn1C.n12ccc(n1)C(=O)N(c1cn[nH]c1)N(CC)CC2.OC N1(C(C2C(C)(C)COCC2)=O)CCOC2(C1)CN(C(=O)C(CCO)N(C)C)C2 c1(C(=O)NCC2(NC(CC=CCC)=O)CCOC2)cc(C(F)(F)F)c(F)cn1 C12(C(N(CCS(C)(=O)=O)C)=O)CCC(NC(=O)CC3CCC3)(CC1)C2 C(=O)(C(O)CCS(C)=O)N(CCNC(c1nc(CC)n(-c2ccccc2)n1)=O)CC c1(CC)ccc(C(=O)NC2C=CC(C(=O)NCC3(O)CCCCC3)C2)cn1 c1(C(N2CC(CCCCNC(C3CC(F)(F)C3)=O)C2)=O)cc2ccccc2c(=O)o1 C1(NC(c2ccc(SC)o2)=O)CCOCC1NC(=O)Cc1nn(C)cc1Cl C(=O)(C(C)(C)CC(C)(C)C)NCCCCC(C)NC(C1CC2CCC1C2)=O N1(C(C(C)SCCCC)=O)CC(CN(C)C(c2cccc(=O)o2)=O)C2(CC2)C1 C(=O)(CCC(=O)N(CC(O)CN(C)C(C1CC(CCO)C1)=O)C)N(C)C c1(C(=O)NCC2CCCN(C(C=CCOC)=O)CC2)cc(=O)n(C)cc1Br Cn1cc(NCC(=O)Nc2cc(CCN3CCCC3)on2)cn1 N1(C(C(CC)F)=O)CCN(C(C2(C3CC3)CC2)=O)CC1CO c1(-c2c(C)n[nH]c2)ccc(F)c(C(=O)NCC(C)N(C(=O)CC(C)C2CC2)C)c1 C1(C(N(C)Cc2ccncc2)=O)CCCC(NC(=O)COc2ccccc2)C1 c1(C(N(CCN(C(=O)CCC(C)(F)F)CC)CC)=O)onc2ccccc12 C1(C(N2C(C(=O)N(CCCN3CCC3)CCO)CCCC2)=O)CCc2ccccc2O1 CCC(O)C(C)(C)C(=O)NCC1C=CCN1C(=O)CCc1cccc(OC)n1 C(=O)(C(C)(C)CCS(C)(=O)=O)N1C(CNC(C2Cn3c(C)cnc3CC2)=O)CC1 C(CC(C)C)(C(=O)NC(C1CC(NC(C2(CO)CCOC2)=O)C1)C)OC c1(CC)ccc(NC(C2(C3CC3)CN(C(C3CC4(CC4)CO3)=O)C2)=O)c(C)c1 C12(CNC(C(CN(C)C)N(C)C)=O)CC1CN(C(=O)C(C)(C)n1cncn1)C2 C1(CCNC(CNS(CC)(=O)=O)=O)CCCN(C(=O)C(C)OCC(F)(F)F)C1 Cc1c(F)ccc(F)c1CNC1CC(C(=O)Nc2ccc(I)cc2C(F)(F)F)C1 c1(C(=O)NCC2CN(C(C(=O)NCC)=O)C2)ccc(C)s1 c1(CCC)nc(=NCOC(=O)OC2CC2)s[nH]1 c1(C(=O)NCC(C)NC(c2c(C)nncc2)=O)cc(C(F)(F)F)ccc1O N1(C(c2ncn(CCNC(C3C=C(C)CS3)=O)c2)=O)CC2CCC(O)C2C1 C(=O)(C(C)C=C=C)N(C(C(=O)NC(C#C)CC1CCCC1)(C)C1CC1)C CC1CN(C(=O)CCC2CC(NC(C3(C)CC3(C)C)=O)C2)CC(C)(C)O1 C(=O)(C(F)(F)C(F)F)N1CC(N2CCN(C(CCCNC(N)=O)=O)CC2)C1 N1(C(c2noc(C)c2C)=O)CC(NC(c2cc(=O)ccn2C)=O)CC(C)C1 C1(CCC)OCCC1C(=O)NCC1CC(NC(c2c[nH]nc2COC)=O)C1 CC1SCCCC1C(=O)NC(CO)C(=O)Nc1cnc(C2CC2)nc1 c1(CN(C(C)C)C)cn(C2CCC(C(=O)NCc3nc(C4CC4)no3)C2)nn1 C1(C(=O)NC(c2ccnn2C)C)COCCN(C(c2cc(Cl)c[nH]2)=O)C1 C(C(CC(C)C)C(=O)N1CCC(C(F)C(=O)NCC2CC3(CC3)C2)C1)OC C1(NC(C(c2ccc(F)cc2)C)=O)CN(C(c2sccc2C#N)=O)C2CCCC12 CC1CN(C(=O)CC2CC2C(F)(F)F)C1C(N1CCC(c2ncco2)C1)=O c12nc(ncc1Cl)CO2.C=C(CNC)CCNC(=O)C(C)NC(N)=O Cn1c(CC(=O)NCC2CC(NC(=O)CC3CC3(Cl)Cl)C2)nnc1S c1(CCC(=O)NCC2N(C(C3C(C)(C)COC3)=O)CCC2)ccc(F)cc1F C#CCC(C(=O)NCC(C)(O)C1CCCC1)NC(=O)CC(C)SC C1(CNC(c2cncs2)=O)CCCCN(C(c2ccccc2OCC2CC2)=O)C1 c1(OCC)nc(Cl)ccc1C(=O)NCC1CC2CCC1N2C(=O)C1=COCCC1 C(C(=O)Nn1ccccc1=O)C12C(CN(C(c3ccc(C)c(C)n3)=O)C1)CC2 Cc1cc(C(=O)NC(C2(O)CN(C(=O)C(c3ccccc3Cl)O)C2)C)ncc1F c1(CCC)cc(C(N2CCC(CNC(c3cc(=O)n(C)cn3)=O)C2)=O)cc(O)n1 C1(C(N2CCC(COCC)CC2)=O)CCCCN(C(C2CC2(C)C)=O)C1 C1(N(C(CCC)=O)CC)CCCN(C(=O)CC2CCCC23CC3)C1 C(=O)(C(F)C(C)CC(=O)OCC)NCC1N(C(Cc2cn(CC)nc2)SC)CC1 CCC(F)(F)CC(=O)NCC1CCC(F)(CNC(c2cc(O)nc(OC)n2)=O)C1 C(=O)(CC(C)(C)NC(=O)CN(C)C(C1CCN1C)=O)NC c1(C(=O)NC2C(CNC(C(C)OCC)=O)CC2)ccn(C)c(=O)c1 c1(NC2(c3n(CCC)nnn3)CC3CC3C2)ccc(Cl)c(CC)c1.C12(CC1)NC2 N1(C(C2C(C)(C(F)(F)F)C2)=O)CC2CCN(C(c3nc4ncccn4n3)=O)C2C1 N1(C(c2ccc(SC)cc2)=O)CC(CNC(c2ccco2)=O)CCC1C c1(OC)cc(C(=O)N(CC(C)CNC(=O)C(C)(C)CN(C)C)C)c(N)cc1F CC(C(=O)NCC(C1CCCC1)NC(=O)C(=O)NCC(F)F)C(C)(C)C c1(C(N2CCCC2CC2CCC2)C(=O)NCCOCC)ccnc(P(C)(C)=O)c1 CCC(CC(=O)NCC1(CNC(=O)C(C)C(F)(F)F)CCC1)C(C)C Cc1cc(NC(c2cnc(-c3cnn(Cc4cccs4)c3)cn2)=O)n(C(C)C)n1 Cc1cc(C(=O)NCC2(F)CCC(NC(C3(C)CC3(Cl)Cl)=O)C2)ncn1 Cc1nn(C)c(C(=O)NCc2ccc(-c3ccco3)cc2)c1Br Cc1cc(Cl)ccc1NC(=O)C(C)N(C1CCN(C(=O)Cc2cc[nH]n2)C1)C CC(CC(N)=O)C(=O)NC(C)(C)CNC(c1ccnc(OC(F)(F)F)c1)=O C12CCCN1NC(=O)N(C)CC(C)NC2=O.CC(C)CC=CC(=O)OC(C)(C)C c1(C(=O)NC2C3(CN(C(C(C)O)=O)C3)CC2)cccc2c1CC(C)(C)C2 CC(C)(CNC(=O)COC1CCCC1)CC(=O)NC1(C)CC1(C)C C1(C(=O)NCCCOCCCCCNC(=O)Cc2cc[nH]n2)(CSC)CCCC1 c1(OC)cc(C(=O)NC2CCCC(NC(=O)CC=C(C)C)CC2)ccc1Cl C1(NC(CCc2ccn(C)n2)=O)CN(C(=O)C=Cc2ccccc2)CC2(CC2)C1 S(=O)(=O)(c1ccccc1C(F)(F)F)N(c1ccnc(N(C2CNCC2F)C)n1)C c1(C(=O)NC(C(C)NC(CSCc2nc(C)sc2)=O)C)cccc(CO)c1C C1(C(=O)NCC2CC(NC(C3COC(=O)O3)=O)C2)Cc2ccccc2O1 c1(C(N(CCNC(=O)C(c2ccnn2C)O)CC)=O)cccc2c1NC(=O)CO2 n1(CCC(=O)NCCC(C)NC(C=CC(C)=O)=O)cnc2cc(F)c(F)cc12 Cc1nn2ccccc2c1C(=O)NC(CO)C(C)NC(=O)C(c1ccnn1C)C N1(C(CCOC)=O)CCN(C(c2cnc(OC)nc2C)=O)C(CCO)C1 N1(C(c2c(OC)csc2)=O)CCC(C(F)(F)F)C(NC(=O)CCOC(C)=O)C1 C1(NC(CCNC(C(C)(C)C)=O)=O)CC2(C1)CC2C(=O)NC1C2CCC1CC2 C(=O)(C(CC1CCC1)NC(=O)CC1(O)CCC1)NC1CC(OCC)C1 C1(O)(C(C(=O)NCc2cccnn2)NC(=O)C(F)c2ccsc2)CCCCC1 C(=O)(C(F)CC(C)(C)C)NC1CCC(CC(=O)NC(c2n(CC)ncc2)C)C1 N1(C(C(CC)n2ccnc2)=O)CCC2(CC1)CC2NC(=O)CC1CCN(C)C1 O=NN1CCCCC1C(N1CCCC1CCNC(c1ccoc1C(F)(F)F)=O)=O c1(C(=O)NC2CCN(C(C(C)NC(=O)OC)=O)C2)ccc2nnn(O)c2c1 C1(C(S(=O)(=O)CC(C2CCC(C)(C)CC2)C)C)CCC(F)(F)CC1 C(=O)(CC(C)C(=O)NC1CC(C(F)C(=O)N(C2CC(F)(F)C2)C)C1)OC N1(C(c2c(C)cnnc2)=O)CC(CO)C2(C1)CN(C(C1(F)CC=CCC1)=O)C2 N1(C(Cc2nc(C)sc2Cl)=O)CC(NC(c2nccn2C)=O)CC(F)C1 C1(NC(C=C(CC)CC)=O)CCSC12CN(C(c1cnc(N)c(N)c1)=O)C2 C1(CNC(CC(=O)NCC#C)=O)CC2CCC(C1)N2C(=O)C(C)CC(C)C Cc1no[nH]c1=NC(=O)C1CCCN(C(=O)CCc2ccc(Cl)c(Cl)c2)C1 C=CCC(CC(C)C)C(=O)N1CCCC1C1(NC(c2c[nH]cc(F)c2=O)=O)CC1 C12(CC#C)CCN(C1)CC1CCN(C1)C2=O.c1(C(=O)OC)ccc(OC)nc1 n1(CC(=O)NC(CNC(C2(F)CC=CC2)=O)C2CC2)nnn(-c2cccs2)c1=O C(c1cc(Cl)ccc1OC(F)F)=CC(=O)NCC1N(C(C(CCC#C)O)=O)CC1 CCC(C)(CNC(=O)CSCCN(C)C)NC(c1csc(S)n1)=O C(CN(C)C)(C(=O)NCCCC)NC(COCCC)=O.C1C(=O)N1 C1(C(N(C)CCc2cccc(F)c2)=O)CCN(C(c2ncnn2C)=O)CC1O c1(C(c2nnnn2C2CCC2)NC2C(CC(C)C)C2)c(Br)n[nH]c1Br c1(C(=O)OC)cc(-c2cn(C3(C(C)(F)F)CC3)nn2)ccc1Cl C(CCCCC(=O)NCC(C)N(C(=O)CCNS(=O)(=O)C(F)(F)F)C)NC(C)=O C1(OC(=O)NC(c2cccc(C(F)(F)F)c2)CC(=O)OC)CCC(F)(F)CC1 c1(C(=O)NCC(C)N(C(c2cnc(=N)[nH]c2)=O)CC)ccc2c(n1)CCCC2 N1(C(=O)OC(C)(C)C)CC2CCC(CNC(=O)CCF)C2C1 CN(C1CCc2cc(Cl)ccc21)C1CCCN(Cc2cc3n(n2)CCCC3)C1 C1(NC(CCC=CC)=O)CN(C(=O)CN2CCC(C)CC2)CCC1O C(=O)(CC1=NNC(=O)C1)N1CCC(CCCCNC(C(N(C)C)C2CC2)=O)CC1 C1(C(=O)NCCC2(O)CN(C(C3C(C)(C(F)(F)F)C3)=O)C2)C2CC3C(C2=O)C13 C1(NC(C(C)SC)=O)CN(C(=O)Cn2ncn(C)c2=O)C2CCCCC12 CC1(C=CC(=O)NCC(F)CNC(=O)Cn2ccnn2)CCOCC1 C1(C(N2C(C(=O)OC)C=CC2)=O)C=CCN(C(=O)C(C)N2CC(C)C2)C1 CCCS(=O)(=O)CC(=O)N1CCCC(COC)(NC(=O)C(C2CCOCC2)F)C1 c1(-c2c(OCC)cc(OC)cc2)n[nH]c2c1CN(C(N1CCC(CO)C1)=O)C2 CC(CN(C)C)CC(=O)NCC1(C)CC(NC(c2cncc(CO)c2)=O)C1 S(=O)(=O)(c1ccc2oc(=O)ccc2c1)N1CC2C(CNC(C(C)(C)Br)=O)(C2)C1 CC1CC(NC(=O)CC(C)(C)c2ccccc2)CN(C(=O)CCc2ccc[nH]2)C1 N(C(=NCCOCCO)N1CCC(C)(OC)C1)CC1C(CCC)C1 CCC(CC(F)(F)F)NC(C1(CCNC(=O)C=Cc2cocn2)CC1)=O N1(C(c2cnc(CC(C)C)s2)=O)CC(CNC(=O)CC2(C(F)F)CC2)C(C)(C)C1 C1(CC(N2CC(C#CC)C2)=O)CN(C(=O)C(C2CCCC2)OCC)C(C)(C)C1 c1(C(=O)NC(C(C)C)CNC(=O)COCC2CC2)cc2cccnc2[nH]1 C1(C(=O)OC)(NC(c2ccc(C3CCOCC3)cc2)=O)Cc2cc(Cl)ccc2C1 C1(C(N2CC3(CCN(C(C(C(C)C)C)=O)C3)C2)=O)CC2CC(O)CC(C1)C2 C1(NC(c2c(C)cc(O)nc2)=O)CS(=O)(=O)C2CN(C(=O)CCC(C)(C)F)CC12 c1(NC(CCOC)C)ccc(S(=O)(=O)NCCc2ccsc2Cl)c(Br)c1 CC(C)(C)C(=O)CCC(=O)N1CCCC(C)(C(N2CCOC(CCO)C2)=O)C1 C1(CCC(C)C)CCCCN1C(=O)NC(C)C(C)(C)C(=O)OC(C)(C)C C1(C(N(CC(CNC(c2c(C)nsc2)=O)O)C)=O)CCCN1C=O c1(N(C(C(CC)C)=O)C)ccccc1-c1cc[nH]n1.C12CCN(C1)C2=O CCC(CCC(=O)N1CC2CC1CN2C(c1cccnc1O)=O)OC CCC(CSC1CCCCC1)(c1nnnn1CC(F)F)NC(C)COCC1CC1 c1(CC2CCC(CN(c3nccc(NC)n3)C)C2)ccc(C)c(C)c1 c1(C(=O)NC2CN(C(CCN(CCCCC)C)=O)C2)c(Br)c(C)nn1C c1(C(=O)NCC2(CNC(Cc3n(C)ncc3)=O)CC2)nnn2c1CCCC2 C1(NC(c2nc(C)oc2)=O)CCN(C(c2ccccc2SCCO)=O)CC1C CC1=C(C)CC(C(=O)NC2CC3(C2)CN(C(=O)COC2CCOCC2)C3)CC1 O=C1Cc2cc(NC3(c4ccc(Br)cn4)COC3)ccc2N1 C(=O)(C(C(C)NC(=O)CCC1(C)N=N1)C(C)C)N(CC#C)CCOC C1(C(N2CC(C)(NC(C3CCN(CC)C3)=O)C2)=O)CCCCN1S(C)(=O)=O c1(CCN=C(NCc2c(C(N)=O)csc2)NCC2CC2)ccc2occc2c1 Cc1cc(C(=O)NC2CCN(C(=O)CN3CC=CC3)CC2C)cc(C)c1Cl c1(OC)cc(C(=O)N(C(C)CNC(C2CCC(C(F)F)CC2)=O)C)c(O)c(Cl)c1 c1(OC)ccc2c(=NCC3CCCC(C)O3)[nH]c(=NC3CC(N(C)C)C3)[nH]c2c1 Cc1cc(C)n(CC(N2CCC(OC3CN(C(c4cnsc4)=O)C3)CC2)=O)n1 N1(C(c2cn(CCCC)nn2)=O)CCN(C(c2nn(C)cc2C)=O)CC1CC c1(OC)ccccc1SCCC(C(=O)NC1CCOC1C)OC(C)C Cc1sc(C)c(C(=O)NCC(C)NC(=O)C(C)NC(c2ccco2)=O)c1C#N N1(C(c2c(CC=C)cccc2)=O)CCC2C(NC(=O)CC3(C)CC(F)(F)C3)CC12 Nc1cc(O)cc(C(N2CCC(n3cc(CCCCCO)nn3)C2)=O)c1Br c1(CC)ccc(C(N2CCC(O)C(C(=O)N(C)C3CC3)C2)=O)c(Br)c1 C1(NC(=O)N(c2ccc(F)cc2)CCO)CCC2(CCC1(F)F)OCCO2 Nc1cccn(CC(N2CCCC(CNC(=O)CCC3CCCC3)C2)=O)c1=O CON(CCC(=O)NC1CCCC1(C)O)C(=O)C1CC(C)(F)C1 c1(C(=O)NC(C2CCN(C(CC=CCC)=O)C2)C)nc(O)nc(O)c1F c1(C(=O)NC23CC(CNC(c4nc(C)oc4)=O)(C2)C3)nnn2c1CCCC2 CN1CCCC(CC(=O)N(C2CCCN(C(c3csnc3Cl)=O)C2)CCF)C1 C1(NC(c2cnc(OCC)s2)=O)CCCN(C(=O)CNC(N)=O)CC1F C1(O)(CNC(c2c(OC)nsc2)=O)CCN(C(C2CCC(OC)C2)=O)CC1 c1(OCC)ccc(C(=O)NC2CCC(CCC(=O)O)C2)cc1Cl c1(CC)cccc(C(=O)NC2CCCC2C(=O)NCCCCOC(C)C)n1 C(CC(=O)N1CCS(=N)(=O)CC1)(C(F)F)NC(c1n(C)ccn1)=O N1(C(CCCOC)=O)CC2CCC1C1CN(C(=O)CCc3cncc(F)c3)CC21 c1(CC(N2CCCC(CNC(C3(C(F)(F)F)CCCC3)=O)C2)=O)ccccc1F C1(N(C(CN2CC(C)C2)=O)C)CCN(C(c2ccc(Cn3cc(Cl)cn3)o2)=O)C1 CCCCC(CC)CC(=O)NC1(CNC(=O)CC(C)c2ccco2)CCCCC1 C(=O)(C1=NOC2(CCC2)C1)N1CCC(CNC(C(c2cc(C)cc(C)c2)C)=O)C1 N1(C(C(C)=CC)=O)C2CCCC1CC(NC(c1ccc(CC(=O)OC)cc1)=O)C2 Cc1ccc(C(C)C(=O)NC2CCC(NC(=O)CCc3nncn3C)C2)cc1 C1(OCC)CC(C)N(CCC2CC=CC2)C(C)C1 c1(CCNC(c2cnc[nH]2)=O)cnc(NC(=O)C(O)CN2CCOCC2)s1 n1(CCNC(C2(CCNC(CN(C)CC)=O)CC2)=O)cccn1 CCC(C)(C)C(O)C(=O)N1CCC2(NC(c3nc(O)ncc3C)=O)CCCC12 CCC(C(=O)N1CCCCC(N(C)C(c2ccc3occc3n2)=O)C1)C(C)(F)F c1(C(=O)NC2CC(N(C(c3c(C)ncnc3C)=O)C)C2)[nH]nc2c1COC2(C)C C1(C(=O)NCC2C(OCC)CN(C(=O)CN3CC=CC3)C2)CC2COCC(C1)C2 C1(NC(c2c(C)cc(C)s2)=O)(CNC(C2CCCC2)=O)CCCCC1C c1(CCC(=O)N(C)CCNC(C2CCCO2)=O)cncc(F)c1 c1(NC(c2nn(CCOCC)c(=O)cc2)=O)sc(C)c(C)c1C#N CC1C(NC(c2cc3occc3[nH]2)=O)CCCN1C(=O)C=Cc1ccccc1 Cc1ccc(C)c(C(=O)N(CCCCN(C(=O)C(C)Cc2ccccn2)C)C)c1 CC1CCN(C(C2(c3cccs3)CC2)=O)C(CNC(=O)C(CCO)N(C)C)C1 N1(C(C(C(C)C)N2CCCC2=O)=O)CC2(CNC(=O)CCOC3CC3)CCC1C2 CC(C)CC(CN=c1ncc2ccccc2[nH]1)N.C1(C(=O)C)CCCCCC1(F)F C1(NC(CC=CC)=O)CCN(C(c2cccc3nnn(C)c23)=O)CCC1(F)F C1(NC(c2nc(C)sc2)=O)CC(O)CN(C(c2n[nH]c(C)c2F)=O)C1 c1(C(=O)NC2C(C=C)CN(C(=O)C(C)O)C2)ccc(S(=O)(=O)C2CC2)cc1 c1(CN=C(NC(C)C)NCc2ccc(S(C)(=O)=O)s2)ccc2ccc(Cl)cc2n1 C1(N(C(C2COCC2O)=O)CC)CCCN(C(=O)C=CCO)C1 CCC(C)C(C)CN=c1[nH]c(=NCc2ccccc2CO)[nH]c2cccc(F)c12 c1(C(=O)NCC2C(C)CN(C(=O)CC3CCCC3C)C2)ccnc(Cl)c1F C#CCCCC(C)C(=O)N(C(C)C(N1CC2CCC(O)C2C1)=O)CC c1(C(=O)NC2CCN(C)C2)cc(Cl)ccn1.C1(C2CC2)(C(=O)C(CCN)=O)CCC1 C1(NC(C(c2ccccc2)C)=O)CCN(C(=O)C(C)n2ccnc2)C1(C)C C=CC(C)(CC)C(=O)N(CCC(=O)NC1CN(C)CC1OC)CC C(=O)(CC(C)(C)C(F)F)N(C)CCNC(c1ncsc1-c1ccccn1)=O C1(C(=O)NC(c2nc[nH]n2)CC)(CC)CCCN1C(c1cnc[nH]c1=N)=O C1(CNC(C2(COC)CC2(F)F)=O)(CNC(=O)CCc2ccco2)CC12CCC2 c1(OCC)cccnc1C(=O)NC1CCCC(CNC(c2cnc(S)nc2)=O)C1 n1(CC#C)cnnc1C(=O)N(CC(=O)NC(C)C(C)(C)C)CCOC CCC(C)CC(C(=O)N1CC(=O)NC(=O)C1)NC(c1n[nH]c2c1COC2)=O c1(CC(=O)NC2(C)CCCN(C(CC(CC)(F)F)=O)C2)cnc2c(C)cccn12 C1(C)(CC)C=C(C(=O)NCC#CCNC(=O)CC(C)c2cccnc2)C1 CC1CCCCC1OCc1cnn(Cc2ccccc2)c1.C1(=O)CCN1CCO C1(C2CC2)(NC(C(CC(C)C)n2ccnc2)=O)CCN(C(=O)Cn2cccc2)C1 N1(C(COc2c(OC)cccc2)=O)CCN(C(C2CCCNC2=O)=O)CC(O)C1 CC1CCCC1(O)n1cc(-c2ccc(N3CCCC3)cc2)nn1 NC(=O)CCCC(=O)NC1CC1NC(=O)CCC(=O)Nc1nccs1 c1(C(C)NC(C2CC(NCC=Cc3ccccc3)C2)=O)cc(Cl)ccc1O CC(C(=O)N1CCN(CC2CN(C(C3(c4ccsc4)CC3)=O)C2)CC1)C(C)O C1(C(N(CC=C)CC2CC2)=O)C2CCCC2CN1C(c1ccc(OC)nn1)=O Cn1nccc1C(C(=O)NC(Cc1ccco1)CO)NC(=O)CCC1(C)CC1 C1(C)(CNC(CC2(CC)CCC2)=O)CCC(NC(=O)CSC(C)C)C1 C(=O)(CC1=CCOCC1)N1CCC(NC(c2c(C)noc2)=O)C1c1ccccc1 N1(C(c2c(CC)occ2C)=O)CCN(C)C(C(=O)NCC2CCN(C)C2CC)C1 c1(C(=O)NCC2(F)CCN(C(Cc3cc(C)on3)=O)C2)ccc(OC(F)F)nc1Cl C1(CNC(C2(OC(C)C)CCC2)=O)CN(C(=O)C2CC2)CC12CC2 N1(C(CC=C)=O)CCC(CNC(=O)C=CCN(C)CC)(COC)CC1 Cc1ccc(C(C)CC(=O)N2CC(CNC(C3C4CCN3CC4)=O)C2)cc1 S(=O)(=O)(c1cc(Cl)cc(Cl)c1O)NC(c1ccc(COC(C)=O)cc1)=O Cc1cc(C(N2CCC(C)(NC(C3CC3C)=O)C2)=O)nn1-c1ccccn1 C1(C)(c2cn(CC3CN(C(c4c(CC)ocn4)=O)C3)nn2)CCCN1C CC(C)C(CO)C(=O)N1CCOCC1CN(C(=O)C(F)(F)c1ccccc1)C Cc1cc(C(=O)NCCn2cc(CNC(=O)Cc3cccs3)nn2)cnc1O N1(C(c2cc(COC)on2)=O)CCC2(NC(=O)CCC3CCCC3)CC2C1 c1(C(N(CC(C)CNC(C2CC23CC3)=O)C)=O)cccc2c1OCCN2C Cc1cc(N(CCC#N)C(c2ccc(Cc3nn[nH]n3)cc2)=O)n2nccc2n1 N1(C(CCCOCC=C)=O)CCCCC(CNC(C2(COC)CCCO2)=O)C1 C=CC1COCCN1C(=O)COC1CCN(C(C2CC3(CCO2)CC3)=O)C1 C(=O)(C(C)CC(=O)NCC1CC(OC)CN1C(=O)CCCn1ccnc1)OC c1(C(=O)NC2C(NC(c3ccc(CC)nc3)=O)CCC2)ccc(C(C)C)cc1F c1(C(=O)NCC2(O)CCCN(C(=O)CC(F)F)C2)n[nH]c2c1CCOC2 Cc1c(C(=O)NCCC(C)NC(c2ncc(F)cc2F)=O)nn(C)c1Br Cc1ccc(C(=O)NC2(C)CCN(CCOC3CCC3)CC2)c(F)c1F N1(C(CNC(=N)N)=O)CCC2(CC1)CN(C(=O)CC1CC1)CCO2 C1(CC)CCN(C(c2nc(Cl)oc2C)=O)C1C(=O)NC(c1cnn[nH]1)(C)C c1(-n2c(C(c3cccc(Cl)c3)Nc3c(C)nc[nH]3)nnn2)ccc(Cl)cc1 c1(SCC)ccccc1CC(=O)NCC1(NC(=O)CC2CCN(C)C2=O)CCC1 CCCCC(O)CC(=O)NC(C)(C)CCC(=O)N(CC(=O)OC)CC1CC1 N1(C(C2C(C)CCN2C(=O)CC2OCCCO2)=O)CC2CC(OC)C(C2)C1 N1(C(CSC)=O)CC2CCOCC2(NC(c2cnn(Cc3ccccc3)c2)=O)C1 c1(C(=O)NC(N2CC(N(C)CC3CCC(C4CC4)O3)C2)=O)ccnc(F)c1F N1(C(c2ccc(OCC)cc2)=O)CCC2C(C1)CN2C(C1CCC1(C)C)=O c1(OC)ccc(COCCCC(=O)NCC=CCNC(C2(C)CNC(=O)C2)=O)cc1 N1(C(C=CS(C)=O)=O)CCC(O)C(NC(c2cccc(N3CCNC3=O)c2)=O)C1 N1(C(Cc2c(C)non2)=O)CC(NC(c2cnnn2C2CC2)=O)CCC1C C1(ONC(=O)C2(C3N(C(=O)CC4CC4C4CC4)CCC3)CC2)CCCC1C#N C1(NC(CCN(CCCCC)C)=O)C2CC1CN(C(c1ccon1)=O)C2 C1(C(=O)NC2(C(=O)NCc3ccc(O)nc3)CCCCC2)CC2(CCOC2)C1 Cc1ccc(O)cc1C(N1CC2CC(N(C(=O)C(C)Cn3cccn3)C)C1C2)=O c1(CCCN(C(=O)Cn2cc(CN3CCCC3)nn2)C)ccc(Cl)cc1 c1(C(C)CC)ccccc1CC1CC(OCC(C)C)C1 CC(C)C(O)CC(=O)NOC(CC(C)C)C(=O)N(C(C)C(C)(C)C)C c1(-c2cn(CC3N(C(=O)CC(Cl)Cl)CC3)nn2)ccc2ccccc2n1 c1(C(=O)NCC2CC(COC)CN2C(C2CC2C(F)F)=O)nn(C)cc1[N+](=O)[O-] N1(C(CN(c2ccccc2)CC)=O)CCN(C(C2CC2(F)Cl)=O)CC1 c1(OC(c2nn3ccc(OC)cc3n2)=O)cc2ccccc2c(Cl)n1 N1(C(c2c(OC)nc(C)cc2)=O)CC2CCN(C(C3CC=CCO3)=O)C2C1C N1(C(CCOCC#C)=O)CCC(NC(=O)CC2CC(OC)C2)C(CO)CC1 c1(C(=O)NCC(C)NC(C2CC2C(C)(C)C)=O)ccc([N+](=O)[O-])n1C C1(C(=O)NCC(CCC)OC)CC(ON=C(C(=O)NC)C)C12CCC2 C1(NC(c2cc(COC)no2)=O)COC2(CCN(C(C3(O)CCCCC3)=O)C2)C1 C(c1cc(Br)ccc1F)=CC(=O)NC(CNC(c1cnn(C)c1N)=O)C1CC1 c1(C(=O)NC(CC)(C)CNC(=O)C(=O)NCC2CC2)cc2ccccc2[nH]1 C(=O)(C1=CC2CCCCCC12)NCCOC(CNC(C1(C(=O)NC)CCC1)=O)(C)C C1(CC(=O)NCCC(C(C)C)NC(C2CCCC(C)C2)=O)CCC2(CCC2)CO1 C1(C(=O)NCC(=O)OC)(NC(=O)CCc2ccc(C)c(Cl)c2)CCS(=O)(=O)C1 c1(CC)ccc(Cn2cc(CC(C)NC(c3ccc(CO)o3)=O)nn2)cc1 C1(NC(C2CC(=C)C2)=O)C=CC(CNC(C2CC=CCO2)=O)C1 c1(OCC)ccc(C(=O)NC2CN(C(c3cc(OC)c(C)nn3)=O)C2)nc1OC c1(C(=O)NCC2CN(C(c3cccc(CC(C)C)c3)=O)C2)cc(F)c(O)c(Cl)c1 C1(C(=O)Nc2c(C)n(C3CC3)nc2)CCN(C(c2csnc2Cl)=O)C12CCC2 CN1CCC(C)(C(=O)N(C)CC2CCCCN2C(=O)COCC2CCOC2)C1=O c1(C(N(C(C)C)CCNC(c2csc(O)n2)=O)=O)c(SC)cnn1C N1(C(C(N2CCOC2=O)C)=O)CCC(C)(C)C1CNC(c1ccnn1C)=O C1(N(C(C(C=CC)O)=O)C)CCC2(CC1)CCN(C(=O)CCCn1cccn1)C2 C1(C(=O)NC2C(NC(=O)Cn3ncc(Br)n3)CCC2)CC2(CC2)CO1 N1(C(c2cc(C)no2)=O)CCN(C(C2(C)CNC(=O)C2)=O)CC1CC1CC1 C1(N(C(c2c(C)nco2)=O)C)CCCN(C(=O)C(F)(F)c2cscn2)CC1 N1(C(CC=CC)=O)CC2CC(CNC(c3ccc(N)cc3C(F)(F)F)=O)C2C1 c1(C(N2C(C(N3CCC(C=C)C3)=O)CC2C)=O)ncnc(O)c1F c1(C(N(CC(=O)N2CCC2)C)=O)ccccc1CN1CCCCCC1 c1(CC(=O)NC(CC)CNC(=O)CCCOc2cccnc2)cc(F)ccc1F c1(C(N2CC=CC(NC(C3CC34CCC4)=O)C2)=O)ccc(C(F)(F)F)c(O)c1 c1(C(=O)NCC(C)(C2CCC2)NC(C(COC)OC)=O)nc2n(c1Cl)CCCC2 N1(C(c2nc(C)n(-c3nc[nH]n3)n2)=O)CCC(O)(C(=O)NCCn2cncn2)CC1 O=C(C(O)C(F)(F)F)NCC1CC(F)(CNC(C2CCO2)=O)C1 n1(C(C)C)ncc(C(=O)NCC2(CNC(=O)Cc3cnsc3)CCCC2)n1 C#CCC(C)(CC)C(=O)N1CCC(=CC(=O)NCCCCCC)CC1 C(C(CC=C)NC(=O)CCN(C(CC)CC)C)NC(CC=CC=C)=O c1(C(=O)NCCC2CCCN(C(C(CC)(C)CO)=O)C2)cc2n(n1)CCN(C)C2 c1(CC(=O)NCC2CCCC2C(N2C3COCC2C3)=O)cccnc1O C1(CNC(c2c(CC)nn[nH]2)=O)C2CN(C(=O)C=CCOC)CC12 C1(C(=O)NCCCCCO)(CC)CCCN1C(c1ncccc1F)=O CCC(CC(=O)NCC1CC(OC)CN1C(=O)CC1COCC1O)OC Nc1ccc(C(=O)NCC2CCC(NC(=O)C=Cc3ncc[nH]3)C2)c(Cl)c1 c1(C(C(=O)NC2CC(NC(=O)Cc3cn[nH]c3)C2)(F)F)cc(Cl)ccc1Cl c1(NC(C2CC2C(N2C3COCC2CC(F)C3)=O)=O)cc(Cl)c(I)cc1[N+](=O)[O-] c1(C(=O)OC)ccc(Cl)c(C(=O)NC(C)(CNC(=O)CCn2ccnc2)CO)c1 CC1(C)CC=C(C(=O)NC2CC(=O)N(C3CN(C(c4ccncc4)=O)C3)C2)CC1 C1(NC(C2CCC2C(F)(F)F)CC)CCC(C(=O)OCc2ccccc2)CC1 c12cccc(c1)CNC(=O)Cc1cn-2nn1.c1(CCN2CCCC2)cccs1 c1(SCC)cccc(C(=O)NCC2CN(C(c3n[nH]c(C4CC4)c3Cl)=O)C2)c1 C(C(CC(F)(F)F)NC(c1ccc(=O)n(C2CC2)n1)=O)NC(=O)Cc1nc[nH]n1 N1(C(CSC(C)=O)=O)CC2CCN(Cc3ccc(I)c(F)c3F)CC2C1 CCCCCCCCCC(=O)N1CC2CC1C2NC(C1CCC2CC2CC1)=O C(=O)(CCCCCNC(c1nnn(C)c1N)=O)NC(CN(C)C)CCO N1(C(C)=O)CCC(c2ccc(NC(=O)C=CS(C)=O)cc2)CC1 C#Cc1cnc(C(=O)NC(C2CCN(C(C3CCCC3(F)F)=O)CC2)C)c(C)c1 C1(CC=C)(NC(=O)Cc2csc(C)n2)CCN(C(C2(n3cnnn3)CC2)=O)C1 C1(O)(C(=O)NCCOCCNC(C(C)Cc2ccncc2)=O)CCC(C)(C)CC1 c1(C(=O)NCC2(NC(CN3CCC(C)C3)=O)CCCC2)ccc2c(c1)COCC2 c1(C(N2CC(NC(CSSC)=O)C(C)CC2)=O)ccn2ncnc2c1 C1(CCNC(c2c(CC)ncnc2)=O)CCCN(C(=O)C(C(C)C)OCC)CC1 N1(CC)N=C(C(=O)N2CCC(C)N(C(=O)C3=C(C)OCCS3)CC2)CCC1=O c1(CC)cc(C(N2CC(OC)C(NC(=O)C(n3nccc3C)C)C2)=O)ccc1F c1(C(=O)NC2(C)CC(NC(=O)C=C3CCC3)C2)cc(F)c(Br)cc1F c1(N(C)C(C2CCCN(C3CCC(c4ccccc4)CC3)C2)=O)ccc(Br)cn1 c1(C(=O)NC2C(NC(COCCCN(C)C)=O)CCC2)nc(O)nc(O)c1F C1(NC(c2n[nH]cc2Cl)=O)CCC(O)CN(C(c2ccncc2F)=O)C1 C=CCC(CC(C)C)C(=O)NC(CNC(=O)Cn1cccnc1=O)CC(F)(F)F C(CC(C(=O)N(C)CC1(F)CCCC1)NC(=O)C(n1ccc(C)n1)C)OCC CCC(CC)CC(F)C(=O)NCC(C)C(F)C(=O)N(C)Cc1ncc(C)o1 C1(NC(Cc2nc(C)[nH]n2)=O)CC12CCN(C(=O)CC1(CO)CC1)CC2 C1(CC)CNC(=O)CN1C(c1c[nH]nc1CNC(C12CC(CO)(C1)C2)=O)=O C=CC(C)(CCOC)C(=O)NC1CCC(NC(c2cc(F)cc(C)c2C)=O)CC1 c1(C(=O)OCC)sc2ncc(CNC(N3CCc4[nH]ccc4C3)=O)cc2c1C N1(c2nc(OC)c(Br)cn2)CCC2(CCCC2C(=O)Nc2cccc(F)c2O)C1 c1(C(C(=O)NCC(CC=C)NC(c2cn3c(n2)CCC3)=O)O)c(C)cccc1C C(=O)(CC1CNc2ccccc21)NCCC1CN(C(CC(C=C)CC)=O)C1 c1(-c2c(C)cc(OCC)c(C)c2)ccc2[nH]cc(C(=O)NCc3nccs3)c2c1 Cc1cc(C(N2CC(CCCCNC(c3cnccc3Cl)=O)C2)=O)c(F)cc1Cl C1(NC(c2cccc(CC)c2)=O)CCC2(CCN(C(=O)C(O)c3ccsc3)C2)C1 C1(F)(C(N(C)CCn2cncn2)=O)CCN(C(c2c[nH]nc2Cl)=O)C1 C(=O)(C(C)(C)C(N)=O)NCCCN(C(=O)CC1CCCN1C)CC C1(NC(=O)Cn2cnnn2)CN(C(C2CC3CC3C2)=O)CCC1F CC1C2C(CCN2C(c2cnc(O)o2)=O)CN1C(=O)Cc1ccccc1Cl c1(C(=O)OC2CCC2CSc2ccccc2)cc(Cl)c(Cl)c(I)c1 C1(C(=O)NCc2c(C(N(C3C(C)CC3)C)=O)con2)CCC(F)(F)C1 C(=O)(CS(=O)(=O)CCO)NCC1N(C(C2C(C)C2C)=O)CC(O)C1 N1(CCC)CCCC(C(C)NC(=O)C(C(C)C)OC)C1 c1(C(N(CCOC)CCNC(=O)C(C)n2cncn2)C)ccc(Cl)c(Cl)c1 C(=O)(C1Cc2ccccc21)NCC1(O)CN(C(c2c(C)cc(Cl)nc2N)=O)C1 N1(C(C(C)OCCCC)=O)CCCC12CCN(C(=O)CN1CCS(=O)(=O)CC1)C2 C(=O)(C1CCC(=O)c2ccccc21)NCC(C1CC1)NC(C(CC)=CCCC)=O c1(CNC(C2(COCC=C)CCCNC2)=O)cc(Br)ccc1I Cn1c(C(=O)NC2CN(C(=O)CCn3cncn3)C3CC23)cc(Cl)c1Cl C1(n2c(C(c3cc(C)[nH]n3)NCC(=O)NC3CC3)nnn2)CCCCCC1 C1(NC(C(CC)OCC)=O)CCN(C(C2CC(F)(F)C2(C)C)=O)CC1CO C1(N(C)C)CCCN(CC(=O)NCC2(C)CCN(C(=O)COCC(F)(F)F)C2)C1 C1(NC(C(c2ccc(C)o2)C)=O)CN(C(=O)CC2(C)CCCO2)CC1C c1(C(=O)NCC2N(C(Cn3ncn(C)c3=O)=O)CC2)ccc2n[nH]cc2n1 C1(OC)CC(CNC(=O)C(=O)N(C)CC2(C)CCCO2)N(c2cc(C)ncn2)C1 c1(C(N(CC(C)CNC(C2CC3CC3C2)=O)C)=O)cc(O)nc2ccccc12 CCCCC(CC)C(=O)N1CC(CC(=O)NC2(C=C)CCC2)(OC)C1 N1(C(C(CCCC)O)=O)CCC2(CC1)CN(C(=O)CC(F)F)CC(C)O2 c1(CN(C(C2(C(=O)OC)CC2C)=O)C)cccc(CNC(c2nnsc2C)=O)c1 CCC(CC)C(C)C(=O)NC1COCCC1C(=O)N(C1CC(C(N)=O)C1)C C1(C(N(C)Cc2cn[nH]c2)=O)CCC(O)CN1C(=O)C(=C1CCCCC1)F C1(C(N(CCNC(c2ccc(CF)cc2)=O)C2CC2)=O)CCC(O)(C(F)(F)F)CC1 C=CCCC(=O)NCC1CCCC1C(=O)NCc1ccc(CO)o1 c1(C(=O)NCC2(C)C(C)CN(C(=O)CC3CCCO3)C2)cc2c(cc1N)CCC2 CC(CC1CCCCC1)C(=O)NCCCCC1CN(C(=O)Cc2cnn(C)c2)C1 c1(C(N(CC=CC(=O)NC(COC)(C)C2CC2)C)=O)csc(C)c1 C1(C2CC2)(CNC(c2cnn(CCF)c2)=O)CCN(C(=O)Cn2cc(Cl)cn2)C1 N#Cc1cnc2ccccc2c1N1CCC(NC(=O)Cc2csnn2)C1 CC(CC(=O)N1CCC(NC(c2cccn2C)=O)C1C)CC(C)(C)C C1(NC(c2c(CCNC(c3c(CC)occ3)=O)n[nH]c2)=O)CN(C)C2(CCC2)C1 c1(CCC)ccccc1NC(C1CCN(C(=O)CSC2CC2)C1)=O C(=O)(C1=NOC(C)C1C)N1CCC(C2N(C(c3c(C)nc(O)[nH]3)=O)CCCC2)C1 c1(N(C)C)cc(C(=O)NCC2(O)CC(NC(C3CCSC3)=O)C2)cc(F)c1 C(=O)(C1=C(C)OCC1)N1CC(SC)C(NC(C2CC3CCC3C2)=O)C1 C1(NC(=O)Nc2ccnn2CC2CC2(F)F)CCn2nccc2C1 c1(C(=O)NCCNC(C2CCN(C(=O)C(O)C3CC3)C2)=O)ccc(C(F)F)cc1 N1(C(c2c(CC)c(C)sc2)=O)CCCC2CN(C(C3(C(=O)N(C)C)CC3)=O)CC12 N1(C(c2occ(C)c2C)=O)CCC(NC(C2CCCC(F)(F)C2)=O)C(CO)CC1 C12CN(C(=O)Cc3cc(F)cc(Cl)c3)CCN1C2.S(=O)(=O)(c1cn[nH]c1)N.CO C1(C(N2C(CNC(C3CCC(CC)O3)=O)C=CC2)=O)CC2CCC1CC2OC C(CCSC)(C(=O)N1CCOCC1CNC(=O)CC=C(Cl)Cl)OC N1(C(C)C)CCOC(C(N2CC(NC(=O)CCc3cncnc3)CC2CO)=O)C1 c1(SC)cc(C(=O)NCC2CC(NC(=O)CC(C)SC)C2)co1 C1(CNC(CC=C=C)=O)CC2CCCC(C1)N2C(=O)CCOC1CCC1 N1(C(c2c(C(C)C)ncs2)=O)CC(NC(=O)CN2CC3CC3C2)C2CCCC2C1 O=[N+]([O-])c1cc2c(nc1O)CN(Cc1nc3cc(F)c(F)cc3[nH]1)CC2 C1(=CC(=O)NCC(C2CCOC2)N(C(C=C(CC)C)=O)CC)CCCC1 N1(C(C(n2c(C)ccn2)C)=O)CC(CNC(C2CCNC(=O)C2)=O)CC(C)C1 C1(C(N2CC(OC)C(NC(c3c(C)ncn3C)=O)C2)=O)CCCNS1(=O)=O CCCCC(C(=O)NCc1ncnn1C(C)C)NC(=O)C(C)SC(C)C Cc1sc(C(=O)NCC2CCCC(CNC(=O)C=Cc3cscn3)C2)nc1O c1(CC)cc(C(N2CC(CC)(NC(C3CC4CCC4C3)=O)C2)=O)cc(O)n1 C=Cn1nncc1C(=O)NCC(CNC(c1ncoc1-c1cnn(C)c1)=O)CO C1(CNC(c2cocn2)=O)C=CCN1C(C1CCCN1C(=O)C1CC1)=O CCC(CC)CC(F)C(=O)NCC1CN(C(c2cnn(CCF)c2)=O)CC1C C1(C(=O)NCC(C)(C2CCC2)NC(C(C)C)=O)CC(c2cccnc2)=NO1 CC1CCC(C)(C(=O)NCCN2CCN(C(=O)CCc3ccccc3F)CC2)C1 C1(C(N(CC(C)C#N)C)=O)(CO)CCN(C(c2cccc(Cl)c2)=O)C1 Cc1snnc1C(=O)NC(CN(C)C)C(=O)N1CCC(NC(N)=O)C1 C(=O)(CCC(N)C(=O)Nc1cn(C)c(=O)nc1O)OC N1(C(Cc2cccc(C)c2)=O)CCCN(C(c2c[nH]c3ccncc23)=O)CC1C CC1C(NC(c2ccnnc2)=O)CC2CCC1N2C(C1CC2CC(C1)C(=O)N2)=O C1(OC)CN(C(c2nn(C)cc2Cl)=O)CC1NC(=O)CC(C)C1CCCC1 N1(Cc2cc(CC)c(C)s2)CC2(C1)CN(C(=O)C(O)CCSc1ccccc1)C2 c1(COC)cc(C(=O)NC2(C)CC(NC(C3(CCCF)CC3)=O)C2)cs1 C1(NC(c2cc(C)[nH]c2)=O)CCCN(C(c2ccsc2C(F)(F)F)=O)C1C CCC(F)(F)CC(=O)N(C(C)CNC(C1CCC1OC)=O)C O=C(Nn1cncn1)C(F)c1ccccn1.C1(c2c[nH]nn2)CC2(CC2)C1 C1(CCC)CN(C(=O)C(C2CCC2)OC)CCN1C(c1cscc1F)=O C(=O)(C(C)OC(=O)C(O)C1CCCC1)N(CCCNCCCOCCO)CC C1(OC)CN(C(=O)CC2(OC)CC2)CC1CNC(=O)CC(c1ccccc1F)C c1(C(=O)NCC(C(C)C)NC(c2coc(S(C)(=O)=O)c2)=O)cc2c[nH]cnc-2n1 Cc1nc(C(=O)NC2CC(O)CN(C(=O)CCOC3CCCOC3)C2)cc(O)n1 C1(CNC(CC(CC)OC)=O)CCCC2CN(C(=O)CCc3csc(=N)[nH]3)CC12 C(=O)(C1=CCC(C)(C)CC1)NC1C(C)CN(C(C2CCc3nc[nH]c3C2)=O)C1 Cc1cc(C(=O)NC2CCC2NC(=O)Cn2ncnn2)c(C)n1C1CCOC1 c1(C(N2C(C)CN(C(=O)CCc3cccs3)CC2)=O)cnn2c1NCCC2 C#Cc1ccc(OCC(=O)NC(CCC)CCCNC(C2C(C)C2C)=O)cc1 C1(C)(C(=O)NC2C(C)NC(=O)CC2)CN(C(=O)Cc2cnsc2)C(C)(C)C1 c1(OCC(=O)NC(CNC(C(C)OCC#C)=O)(C)C2CC2)cccnc1Cl C1(NC(C(C)OCC#C)=O)CN(C(=O)C=CCn2cncn2)CC1OC C(=O)(C(CC1CCCO1)C(F)(F)F)NCC1(NC(=O)CC=C(Cl)Cl)CCOC1 c1(C(=O)NC(CN(C(=O)CC(n2nc(C)cc2C)C)CC)C)c(OC)noc1C N1(C(COC)=O)CC(CNC(=O)C(C)NC(C2CCC2)=O)CC1(C)C CC1Cc2cc(CNC(c3noc(-c4ccc(Cl)cc4)n3)=O)ccc2O1 c1(C(=O)NC2(COC)CC2)cccnc1NC(=O)C(C)NC(=O)CC1CCCC1 C1(N(C)C(C2CC(=O)N(C3CCCC3)C2)=O)CCCCN(C(=O)C2=C(Cl)CC2)C1 C(=O)(CN=c1cc[nH]cc1)NCCC1CCCN(C(CCC=C)=O)C1 CC1CC(NC(=O)CNC(C2CCC2)=O)CN(C(=O)Cn2cnc([N+](=O)[O-])c2)C1 c1(CC)c(C(=O)NC2COCC2CNC(C2CCC(O)CC2)=O)cnn1CC N1(C(C(CC(C)C)OC)=O)CC2CCN(C(=O)COC(F)(F)C(F)(F)F)C2C1 S(=O)(=O)(c1cccc2cccnc12)NC1CN(C(c2cncc(Br)c2)=O)C1 C1(CC(=O)OC)(CNC(=O)Nc2ncc[nH]c2=O)CCCCC1 C1(C(N2CCC(N(C(C3C(OC)CC3)=O)C)C2)=O)CCc2nc(C)[nH]c2C1 N1(C(C2CC(C)OC2)=O)CCCCC1C1CCN(C(c2ccnn2CC#N)=O)C1 Cc1ccc(C)c(C(N2C(CNC(C3(CN(C)C)CC3)=O)CC3CC23)=O)c1O c1(C(N(CCNC(C2C(C)CC2)=O)C2CC2)=O)cc(C2(C)CC2)n[nH]1 CCCC(C)(C)CC(=O)NCC(C)(C1CCC1)NC(=O)CC1(C)CCCC1 C(=O)(C(C)CCCC(C)=O)NCC(CCC)C(N1CC(F)(F)C(F)(F)C1)=O c1(OC)ccc(CN(C)C(=O)NC(C)Cn2ccnc2)c2ccccc12 CS(=O)(=O)c1sccc1CNCc1cc(I)cs1 N1(C(CCCCC)=O)CCCC(C2(NC(c3cc(C4CCC4)[nH]n3)=O)CC2)C1 N1(C(C(CC)SC)=O)CCC(C(=O)N(C)C(C2CCOCC2)C)=C(F)C1 C1(C(=O)NC2CC(COC(F)(F)F)C2)CCCCN1C(c1ccc(O)nc1)=O C1(CC(=O)N(C(c2cccnc2)C)C)CN(C(=O)CC2(C)CCCCC2)CCO1 Cc1nc(F)ccc1-c1cn(C2CCN(c3ccccc3)C2)nn1 c1(CC(N2CCC(CCOC)(NC(=O)C(F)OC)C2)=O)c(C)cccc1F N1(C(C2C(CCC)C2)=O)CCC(N(CCC)C(c2ccc(OC)cc2)=O)CC1 CCCCC(O)C(=O)NC1CC12CC(NC(=O)Cc1sccc1C)C2 CN1CCN(C(=O)C(C2CCCO2)NC(c2cccc(O)n2)=O)C(CCO)C1 c1(C(=O)NCC(c2ccccc2)NC(C(COC)OC)=O)nc(Cl)oc1C c1(OCC)ccc(NC2(c3nnnn3CC)CSCC2C)cc1 c1(C(N(C2CC(NC(C3CC(=C(F)F)C3)=O)C2)C)=O)ccc([N+](=O)[O-])o1 C(CC(C)(O)C(=O)NCC1CCN1C(C1COCC1(C)C)=O)N(C)C c1(OC)nc(N2CCOCC2CC(N2C3COCC2C3)=O)ncc1Br C=CC(C)C(C)C(=O)Nc1cccc(NC(c2cc(Cn3cccn3)on2)=O)c1 c1(C2(NC(N(CC)Cc3csc(C)c3OC)=O)CC2)ccc2c(c1)OCO2 CC(C)(C(O)C(=O)N1CCC(Nc2ccccc2Cl)C1)c1ccc(Cl)cc1 C1(C(N2CCN(C(CNC(CS(C)(=O)=O)=O)C(F)F)CC2)=O)CC12CCOCC2 C1(NC(c2c(CC)scc2)=O)(COC)CCN(C(=O)Cc2c(Cl)cnn2C)CC1 c1(C(=O)NC(CCOC)CNC(C2CC=CCC2)=O)c[nH]c(=N)c2[nH]ccc12 N1(C(C2CCCN(CCC)C2)=O)CCC(NC(c2nccn2C)=O)C12CC2 C1(CC(N2CC(F)(CNC(C3CC(SC)C3)=O)C2)=O)CC(C)(C)C(=O)N1 Cc1cccc(C(=O)NC(C)(C)CC(=O)N2CCC(CC(N)=O)C2)c1N C(=O)(CCCCC(N)=O)NCC1C(NC(c2cc(OC)no2)=O)COC1 C1(C2(O)CN(C(c3c(C)nn(C)c3Cl)=O)C2)(CNC(C(C=C)C)=O)CC1 C(=O)(C1=CCCC1C)NC1CC(CC(N2CC(C(CC)CC)C2)=O)C1 S(=O)(=O)(c1cc(Br)nn1-c1ccccc1CSc1ccccc1)N1C(C)CSCC1 C1(N(C(c2cnc(C)[nH]2)=O)C)CN(C(c2ccc(F)c(Br)c2)=O)CC12CC2 Cc1ccc(CSCC(=O)N(C(C)CCNC(=O)C2=COCCC2)C)cc1 N1(C(c2ccc(COC)[nH]2)=O)CC(CNC(C2CCN(C(N)=O)CC2)=O)CC1C C1(C(N2CCC(O)(C(N)=O)C2)=O)CC2(CC(NC(=O)CSc3nc[nH]n3)C2)C1 C1(NC(C2CN(C)C(=O)C2)=O)CN(Cc2ccc(N(C)C)c(Cl)c2)CCC1O C=C=CC(C)C(=O)NC(CNC(C1CN(c2ncc(F)cn2)C1)=O)CC=C c1(NC(C2C3CC2N(Cc2cnc(Cl)c(F)c2)C3)=O)cc(Br)ccc1O C1(CCNC(c2occc2Cl)=O)CC(F)(F)CN1C(c1cc(O)nc(O)n1)=O c1(OCC)cccc(NC(=O)C(c2ccc(OC)cc2)N(CCOC)C2CC2)c1 C(=O)(C(C)CC(C)C)N(C(=O)CC1C(NC)CC1O)CC=Cc1ccccc1 C1(NC2(c3nnnn3CC3CC3)CC(C=C)C2)Cc2ccccc2C1 c1(CCOC)cccc(CN2CCCC(C(N3CCC(F)(F)C3)=O)C2)c1F C(CCCO)N(C(=O)C(C1CC1)N(CCOC)CC)CCCOCC CC(C)C(CNC(=O)C(O)CCNC(=O)CN1CCC(C)CC1)CO C(C(C(=O)Nc1cnn(C)c1)NC(=O)CCc1cccnc1)OC(C)C c1(C(N2CC(N(C(C(C)Cc3cnc[nH]3)=O)C)C2)=O)ccc2nc(O)oc2c1 N1(C(CN2C(C)CCC2)=O)Cc2n[nH]cc2C1C(=O)N1CC(c2ccon2)C1 Cn1cccc(C(=O)NC2CCCC2NC(c2cc(Br)ccc2O)=O)c1=O CCC(CC)(CN=c1cc(C(C)C)nc(Cl)[nH]1)NC(=O)Cc1ncccc1C C1(NC(CCCCC)=O)CN(C(c2cccnc2NC)=O)C2(CCC2)C1 N1(C(c2c(OC)ccs2)=O)C2CCC1C(NC(=O)C(C)CN(C)C)C2 C1(C(=O)NCCCN(CCCCNC(=O)C2CC2)C)CC(O)C12CCC2 c1(C(=O)NCCCn2cc(C3CCN(C)C3)nn2)c(F)cccc1[N+](=O)[O-] Cc1c(C(=O)NCC23CC(NC(=O)C=Cc4cnc[nH]4)(C2)C3)[nH]c2ccccc12 C1(NC(C(Cc2c(C)nc[nH]2)O)=O)CCCC(NC(c2cccs2)=O)C1 C1(COC)CCCN(c2nnnn2Cc2csnn2)C1 C12(NC(COCCC#C)=O)CCCN(C(=O)C(CC)OC3CCCC3)CC1C2 c1(CC(=O)NCCC(C)N(C)C(C2CC23CC3)=O)c(Br)ccc(F)c1F C1(=O)C(C(C)(C)C)n2cc(nn2)N1.C(C(C)CC(=O)N1CCOC(CO)C1)OC c1(C(=O)OCC)ccc(NCC2CN(C(c3ccc(NC(C)=O)nc3)=O)C2)cn1 N1(C(c2cn(CC=C)nc2)=O)CCC(C)C(N(C(=O)Cc2n[nH]c(=N)s2)C)C1 Cc1ccc(C2CC2C(=O)NCCNC(C2CCC(c3ccccc3)C2)=O)cc1 c1(CC(=O)NC2CCCN(C(=O)Cn3nnnc3C3CC3)C2)c(O)ncnc1O C1(C(NOCC)=O)CC12CCN(C(c1cnn(C)c1OC)=O)C2 C(=O)(C(O)CC(C)C)NCC(CC=C)NC(c1ccc(=O)n(CC)n1)=O C(=O)(C(C)C(O)CC(C)C)NCc1occ(C(=O)NC(CC#C)CO)n1 C1(C(N2CCC(C(C)NC(CN3CCC(C)C3)=O)CC2)=O)CN2CCCC2CO1 C(=O)(CCCC(=O)NC1CC(C)N(C(C2CCCC2C)=O)C1)NC N1(C(C2N(C(c3cc(OC)no3)=O)CCC2)=O)CCc2nn(C)cc2C1 C1(C(=O)OC)CC2(CC2)CN1C(C1CC(F)CN(C(C2(Br)CC2)=O)C1)=O CC1CCC(C)N1CC(=O)NCC1CCCCN1C(C1CC1C(C)O)=O CCC(C(C)CN(C)C)NC(C1(NC(=O)CCn2cncn2)CSC1)=O c1(C(C(=O)NCC(CC)(C)NC(=O)Cc2csnn2)O)ccc(OC)cc1 N1(C(C2CN(CC)C(=O)CC2)=O)CC2CC1CN(C(C1C(F)(F)C13CCC3)=O)C2 C12(C(=O)NC(c3c(C)n[nH]c3C)C)CCC(NC(C3CC3C3CCC3)=O)(CC1)C2 c1(N2CCC(O)(C(C)NC(c3c(CC)nco3)=O)C2)cc(C)c([N+](=O)[O-])cc1Br c1(CNC2CCCC(C(=O)Nc3cn[nH]c3)C2)c[nH]c2ncc(Cl)cc12 c1(OC)cccc(C2CCCN(C(=O)CCc3cn(C)nc3C)C2)c1F CC1(C)CCCOC1CC(N1CCCCC(CNC(c2n[nH]c(O)n2)=O)C1)=O n1(CC)cc(C(C(=O)NCCC2CC2)N(C2CC2)CC2(C)CCC2)c(C)n1 N1(C(CCSC)=O)CCOC2(CCN(C(C3(F)CCOC3C)=O)C2)C1 Cc1cccc(C(=O)NC2(CO)CCN(C(C3CN4CCN3CC4)=O)CC2)c1O c1(-c2c(C(N3CCC(NC(CN)=O)CC3)=O)cccn2)nc2ccccc2o1 C1(NC(N(CCCn2ccnc2CC(=O)OC(C)(C)C)C)=O)C2CC3C(C2)C13 N1(C(C2CC3C(C2)C3(F)F)=O)CC2CCC1C(C(=O)Nc1cccnc1)C2 CCCCCC(O)CC(=O)N1CCCN(C(c2ccc(O)c(C(N)=O)c2)=O)CC1 c1(C(=O)NCC=C2CCN(C(CC=C)=O)CC2)cc2c(Br)coc2cn1 c1(C(=O)OC2C(CC)CN(C(=O)NC)CC2)cc(OC)c(OC)cc1CC(C)(C)C Cc1sc(C(N2CCC(F)(CNC(c3cc(C(F)(F)F)c[nH]3)=O)C2)=O)c(C)c1C c1(C(C(=O)N(CC(C)NC(=O)C(F)(F)CO)C)(C)C)c(F)cccc1F C12(NC(C=CC(=O)N(C)C)=O)COCCC1CN(C(=O)COC1CC1)C2 C12CC(=NO1)C(=O)N2.C12(NC(C(n3c(C)ncc3)C)=O)CC1CN(C)C2 Cc1cc(C)c(C(=O)NCC2CN(C(=O)C=CC(=O)N(C)C)CCC2C)cc1C Cc1cncc(C)c1C(=O)NC1CC1NC(=O)C(F)(Cl)c1ccccc1 c1(C(=O)NCC2CN(C(C3CCN(CC)C3)=O)CC2O)cc2c[nH]cnc-2n1 N1(C(C2C(C(=O)OC)C2)=O)CCC2CN(C(c3c(SC)cccc3F)=O)CC12 CC1CC(C(=O)NC2(CNC(c3cncc(N)c3)=O)CCCC2)CC(C)(C)C1 c1(N(C(=O)CC(C(C)(C)C)Sc2ccc(-c3ccccc3)cc2)C)ccc([N+](=O)[O-])cc1 CC(C)(C)CCC(=O)N1CC(CCCCNC(c2cocc2Br)=O)C1 N1(C(Cc2c(Cl)cn(C)n2)=O)CCCC(NC(=O)CCOC2CCOC2)CC1 CCC(CN(C)C)CC(=O)NCCc1cc(C(=O)NCc2cccc(F)n2)no1 c1(CN2CCC(NC(c3cncc(CC)c3)=O)C2)cc(C)cc(Br)c1 c1(C(N(CC(=O)NCCC(C)O)CC#C)=O)oc(C)nc1C c1(CC(N2CC3C(CNC(CCCCCOC)=O)C3C2)=O)ccc(S(C)=O)cc1 O=C(C1CCCc2nn[nH]c21)NC1CCSC12CN(C(C1(CO)CCCC1)=O)C2 C#CCC(C)(C(=O)NOCCCOC)NC(c1ncncc1N)=O c1(OCC(N2C(C(=O)OC)CC2)=O)ccc(Cl)c(Cl)c1 c1(C(=O)NC2(C)CCN(C(C(c3ccc(C)s3)C)=O)C2)n[nH]c2c1CC(C)(C)C2 c1(C(=O)NC(C)C(CO)NC(C2CC(F)CN2C)=O)cn2ccc(F)cc2n1 c1(OCCC(=O)N(C2CCN(C(C3CC34CC4(F)F)=O)C2)CC)ccc(C)cc1 c1(OC)ccc(C(=O)NC2(C3CCCN3C(C3C4CCCCC34)=O)CC2)cc1 C1(C(N2CCC(N(C(=O)Cc3nc[nH]n3)CCO)CC2)=O)(OC)CCCCC1 N1(C(c2cc(CCCCC)[nH]n2)=O)CC2CCN(C(C3CCCN(C)C3)=O)CC12 N1(C(C2CN(C(CCCCCC)=O)CC23CC3)=O)CCC(C2CC2)CC1 c1(C(=O)NCC2CC3CC3N2C(=O)Cc2ccnc(Br)c2)cc(F)c(F)cc1O Cn1ccc2sc(C(=O)NC3CN(C(=O)Cc4c[nH]nc4O)C3)cc12 Cc1cc(CN2CCC(N)C(C)C2)c(O)c(Cl)c1 c1(C(=O)NCC(CC=C)NC(=O)CC2C=NN(C)C2=O)ccc(CC)cc1O C(=O)(C(C(=O)NCCCOC1(C(N(C)NC(=O)C2CC2)=O)CC1)C1CC1)OC C(=O)(C(C)(CO)NC(c1cccnc1S)=O)NCC(COCC)C C1(NC(C(F)=CCC)=O)C2CC3CC(C2)CC1(CNC(C1(S(C)(=O)=O)CC1)=O)C3 C1(c2n(C)ncc2)CN(C(c2cc[n+]([O-])cc2)=O)CCN1C(=O)CNC(N)=O C(=O)(C(F)C(F)(F)F)N1C(C)CC(NC(=O)COc2ccccc2Cl)C1 N1(C(C(C)(C)NC(c2cncc(C#N)c2)=O)=O)CC2CCC1C(O)C2O N1(C(c2c(C)noc2)=O)CCC2(CCOCC2)C(CNC(=O)C2=CCCSC2)C1 C1(C(=O)NCCC(=O)NO)CCOCC1NC(C1CC1(Cl)Cl)=O N1(C(C(CCC)F)=O)CC2COCC2(C(=O)NC(CC(C)C)C(=O)OC)C1 N1(C(C(C)C)=O)CCN(C(c2cccc(C(=O)C3CC3)c2)=O)CCC1C c1(NC(C2CC23CCN(C(=O)CC2CCC2)C3)=O)cnc2ccoc2c1 N1(C(C(n2c(C)ncc2)C)=O)CCC(C(=O)NC2(CCO)CCC2)C12CCC2 c1(C(=O)NC2CC(C)(NC(c3c(COC)nn(C)c3)=O)C2)c(Cl)ccc(O)c1N N1(CC(NC(=N)NCCc2nccs2)C)CCCCC1 c1(C(C)C)scnc1C(=O)NCC(O)CN(N1CCOCC1)C(C1CCNC1=O)=O c1(CC)c(C(=O)NCC(C)(CC)NC(C2CC3CCC2C3)=O)csc1C S(=O)(=O)(c1ccc(N2CCSCC(C)C2)c(F)c1)N(CC(OC)OC)CC(C)C c1(C(=O)NC2C(C)(OCC)C2)cc([N+](=O)[O-])cc(I)c1C N1(C(c2cn(CCC(C)(C)C)nn2)=O)CC2CC1CN2C(=O)CCCF N1(CCC(=O)NCCCCC(C)NC(CCCC(=C)C)=O)Cc2ccccc2C1 c1(CNC(CCC=C)=O)ccc(N2CCN(C(C3(SC)CCC3)=O)CC2)cc1 c1(OC)cc(NC(c2nc(C(=O)NCC3(C)CCC3)cs2)=O)ccc1O C(C)(C)(CC(F)C(=O)N(C1CSC1)C)NC(CC(COC)(C)C)=O CC(C)CC(O)C(C)C(=O)N1CC(CNC(=O)CCSCC(C)C)C1 c1(OC(C)C)ccc(C(=O)NC2CC2C(=O)NCc2ccc(Br)nc2)c(F)c1 C1(CC)CCCC(CNC(=O)CCCNC(c2ccccc2NC)=O)C1 c1(C(=O)NCC2C(CC(=O)NC3C(C)CCC3)C2)cnn2c1OCC2 Cc1nn(CC(=O)NC(C)CCNC(C2CCCN2c2nccs2)=O)c(C)c1C C1(C)(C(=O)NCC#CCNC(COCCN(C)C)=O)Cc2ccccc2C(=O)O1 C(=O)(C(Cc1ccco1)CC(C)C)N(C1CCC(NC(=O)C2=COCC2)CC1)CC N#Cc1cc(NC(C2CSCCN2C(c2cc(F)ccc2Cl)=O)=O)cc(F)c1F N1(Cc2cnc(C)s2)CCC(NC(c2ccccc2OCC2CC2)=O)C(C)C1 CC(C)C(C)C(=O)N(C1CCCCC1N(C(=O)CSc1cnn(C)c1)C)C Cc1ncc2n1CCN(C(=O)CC1CCC(NC(c3cn(C)c(=O)n3C)=O)C1)C2 Nc1c(C(N2CCC(NC(c3cc[nH]n3)=O)C(F)C2)=O)cnc2ccnn12 C1(C(N(CC(=C)C)C)=O)CCN(C(=O)C(n2cc(C)cn2)C)CC1(C)C N1(C(C2C(C)(C)CO2)=O)CC(NC(=O)CCc2cccc(O)n2)C2(CC2)C1 CC(O)CCCN=c1[nH]c(=NCC2CC23CCC3)c2c(F)cccc2[nH]1 c1(C(=O)NC2CCN(C(C3C(COC)C3)=O)C2)c(O)cc(Cl)cc1Cl CC1=NOC(=O)C1CC(=O)NC(C1CCN(C(C2C3CCCC23)=O)C1)C C1(NC(C2CC(CC)OCC2)=O)CC2(CCCCN2C(=O)CCOCC(F)F)C1 C1(C(N2CC(CCNC(c3c(COC)n(C)nc3)=O)C2)=O)CCOCC12CCC2 c1(C(C)NCc2ccc(F)cc2Cl)cc2cccc(F)c2o1 N1(C(CN2CC(C)C2)=O)CCN(C(=O)C(c2cccnc2)C)CC1CO C1(CC)CCCN(C(c2cc(C)[nH]n2)=O)C1C(=O)NC1COC2(CCC2)C1 c1(C(=O)NCC(CO)NC(CC(CCCCC)O)=O)cccc2c1NC(=O)CC2 C1(C(N(CCC(=O)N(CC(Cl)Cl)C)C)=O)CC(C)(C)CCO1 c1(CNC(N2CCOCC2c2nc[nH]n2)=O)ccnc(F)c1F CC(C)CC(C)C(C(=O)Nc1ccc(F)cc1)N1CCC(NC(=O)C(C)C)CC1 N1(C(c2oc(C)c(Br)c2)=O)CCN(C(c2ccc[nH]2)=O)C(CC(F)F)C1 C(C(C)N=c1ccnc(CO)[nH]1)(C1CCCCC1)NC(CC(CCC)O)=O N1(C(C(CC)C(C)C)=O)C2CCC1CC(CNC(=O)Cc1cnnn1C)C2 Cc1cn2c(n1)C(C)CC(C(N1CCCC1C(C)NC(c1csnc1C)=O)=O)C2 N1(C(C(C)(C)c2cnco2)=O)CCC(C)(NC(=O)Cc2sccc2Cl)C1 c1(OC)ccnc(C(N2CCOC(C(=O)Nc3cncc(Cl)c3C)C2)=O)c1OC C1(CNC(C(C)C(C)(C)C)=O)CC2(CCN(C(c3cc(F)ccc3Cl)=O)C2)CO1 c1(C(=O)NC2CC3CN(C(C4(OC)CC4)=O)C2C3)cc(S(C)(=O)=O)oc1C n1(CCOC)cc(CN2CCC(NC(=O)C(C)OCC)C2)nn1 C(=O)(C(O)C(C(C)C)OC)N1CCCC(C(N(CC(COC)O)C)=O)CC1 C1(NC(c2cccc(=S)n2O)=O)CC12CCC(NC(=O)C(F)n1cccn1)CC2 c1(C(=O)NCC(C)N(C(=O)Cc2ccnc(F)c2)C)cc(=O)c2ccccc2o1 c1(C(=O)NCCC2C(C)(C)C2)cc(OC2CCCC2)ncn1 CC1CCCCC1CC(=O)NCCOC1(CNC(=O)CS(N)(=O)=O)CCOCC1 Cc1cc(F)ccc1CC(N1CCN(C(C2CCCN2C=O)=O)CC1C1CC1)=O C(=O)(CCCCCF)NCc1ccc(CC(C)NC(Cc2c(C)non2)=O)cc1 n1(CC(=O)NC2CCCC(CNC(C(C)NC(C)=O)=O)C2)ccc(=O)cc1C c1(SC)cccc(C(=O)NCCC(O)CNC(c2cc(C(N)=O)c[nH]2)=O)n1 c1(C(N2CC(NC(C#CC(=O)O)=O)C(O)C2)=O)cnc2cc(Cl)ccn12 C(C(=O)NCCC1CN(C(=O)CN(CCO)CCO)CCO1)(C(C)C)SC c1(C(=O)NC2CCN(C(c3cc(C(N)=O)oc3)=O)C2)ccnc2ccncc12 C12CC(O)CN1C2=O.C(=O)(C(O)C(F)F)N(C)CCCO.N12CCC(CC1)C2=O N1(C(C2(OC)CCC2)=O)CC2(CCN(C(c3ccc(F)c(F)c3C)=O)C2)C1 C1(CC)(CNC(=O)C=C(C)Cl)CCN(c2cc(C)nc(-c3ccccn3)n2)CC1 C1(C(=O)NCCN(C(=O)CC2CCCC(C)(C)O2)C)C2CC(F)(F)CC12 Cc1cnc2nc(C(=O)NCCCCN(C(=O)C(C(C)C)NC(N)=O)C)nn2c1 c1(C(=O)NC2CCC(N(C(c3cc(OC)no3)=O)C)C2)cccc2occc12 N1(C(c2c(C)nccn2)=O)CCC(CNC(C23CC(CO)(C2)OC3C)=O)C(C)C1 O=C(CS(=O)CCC(F)(F)F)N1CC2CCN(C(=O)COCCF)C2C1 CC(C)(C)C(C(=O)NCCNC(C1CCCO1)=O)n1ccnn1 N1(C(C2N(C(CC(C=C)C)=O)CCCC2)=O)CCOC2COCC2C1 c1(C(N(C2CCN(C(=O)CSC)C2)CC#C)=O)cc(C(C)C)oc1C(C)C C=CCN(OC)C(=O)C1(NC(=O)CCCCCF)CCC1 C1(C(C)(C)C)CCC(CO)N(C(=O)CC2(CC(=O)O)CC2)C1 c1(CNC(CCOCC)=O)ccc(C(=O)NCC(c2cccs2)C2CCOC2)[nH]1 c1(C(N2C(CNC(C3(C)ON=C(C)C3)=O)C(C)(C)CC2)=O)c(C)nc(C)nc1C C(CCC(C)C(=O)NCCOCCOCCOCCN(C)C)OC.C1CC(=O)N1 N1(C(C(C)CN(C)C(c2coc(N(C)C)n2)=O)=O)CCC(C)(C)C(CO)C1 c1(C(N2C3CN(C(C(CC)=O)=O)CC2C3)=O)ccc2c(c1)NCC(=O)N2 C1(NC(=O)CCc2ccc(Cl)s2)CC(NC(C2CC3CCC2O3)=O)CC1O CCCCC(C(=O)NC(C)CCNC(c1ccc(C(C)=O)[nH]1)=O)N(C)C CCCC(C)C(=O)NCC(c1cccc(Cl)c1)NC(=O)CCN1CCOCC1=O C1(CC(=O)NC2(COC)CN(C(=O)CCC(=O)N(C)C)C2)C(=O)N(C)N=C1C C(=O)(CC(C)(C)NC(=O)C(C)(C)F)NCCC1(COC)CC1 N1(C(CC(C(C)O)N)=O)CCCC(C2CC2NC(=O)C(F)(F)F)C1 Cn1nc2ccccc2c1C(=O)NCC1(NC(C2CC2(F)Cl)=O)CCCCC1 C1(CNC(CC=C)=O)CC2CCC(C1)N2C(C1CC(C2CCCC2)C1)=O Cc1cc(C)n(CCC(=O)NCCC2CCN(C(C3C(F)(F)C34CC4)=O)C2)n1 C1(NC(C2(C)CCNC(=O)C2)=O)CC2(CCN(C(C3(F)CCC3)=O)C2)C1 C1(NC(C(C)n2ccnn2)=O)CCC(F)(CNC(=O)CN(C)S(N)(=O)=O)C1 N1(C(C(C)OC)=O)CC(CNC(=O)CC(=O)NCC(F)(F)F)C2(CC2)C1 CC#CCC(C(=O)NCCN1CCCCC1)NC(=O)CN(C)C(N)=O C(CCC(=O)NCC1(C)CC(NC(=O)C(F)n2ccnc2)C1)SC c1(C(=O)NC(C)Cn2cc(CCCO)nn2)ccnc(-c2nccs2)n1 C1(CC=C)(NC(C2(C)CC2c2ccccc2)=O)CCN(C(=O)C(CC)OCC)C1 c1(C(N(C2CC(NC(=O)CC3SC(=N)NC3=O)C2)C)=O)csc2c(O)ccnc12 c1(CNCC23CCCC(C)(OC2)C3)cccn2c(C(=O)O)cnc12 C1(NC(C=C(CCN(C)C)Cl)=O)CCN(C(=O)CC2CSC2)CC12CCC2 CC1(C)CC(NC(=O)CCN(C(=O)CC2CCCC23CC3)C2CC2)CC(O)C1 c1(OCC(=O)OC)cccc(CCC(C)NC(=O)C(=O)NCC2(C)OCCO2)c1 C12(C(=O)NC3CC(NC(=O)CCCCCn4cnnn4)C3)CCCCC1OCC2 c1(C(=O)NCCC(CCNC(c2c(C)con2)=O)C)cc2c(O)ncnc2cn1 CON(CCC(=O)NCC(N1CCCCC1)=O)C(=O)C1CCN(C)C(=O)C1 C1(C(N2CCC(CNC(C(CCC)C)=O)(OC)C2)=O)CS(=O)(=O)CC12CC2 Cc1csc(C=CC(=O)NC(C2CCN(C(c3nc(Cl)oc3C)=O)C2)C)n1 Cc1nn(C)c(C)c1C(=O)C(N1CCC(NC(c2scnc2C(C)C)=O)C(O)C1)=O N(C(=NCCC1(C)OCCO1)NC(C)C)C1CC(OC)C1(C)C C1(C(=O)NC(C(C(=O)OC)C)C)C(C2CC2)CCN1C(C1CCC1)=O c1(C(=O)NC2CCC(NC(=O)C(O)Cc3cnc[nH]3)C2)ccn2c1CSCC2 C1(C(=O)NCCN(C(=O)CCCCC2CC2)CC)CN2CCN1CC2C CC1=NC(C)(CNC(=O)C(C2(O)CCC2)NC(C2C3CCC(F)C23)=O)CS1 N1(C(Cc2cc(COC)on2)=O)CCOCC1CN(C)C(c1cscc1Cl)=O CC1CC=CCC1C(=O)NCC1CCN(C(=O)CCCc2cccc(Cl)c2)C1 c1(CNC(N(C)CP(C)(C)=O)=O)cc2c(cn1)CCCC2 C1(C(=O)NC(CC=C)CNC(=O)CCn2cccn2)CC2(C1)CC21CC1 N1(C(=O)Cn2ccccc2=O)CCC2CCC(C1)N2C(C1CCCCC12CC2)=O c1(C(=O)NCCC(C)NC(=O)C(O)CF)cnn(CCO)c1 C1(NC(C(F)=C(C)C)=O)CCC2CN(C(c3cncc(N)c3C)=O)CC2C1 C1(NC(C=C(C)Cl)=O)CCCCC12CCN(C(C1(F)CC3(CCC3)C1)=O)C2 CC1(C(=O)NCC(N2CCC2)C2CC2)C=CCN1C(C1CCC1)=O C1(CC(=O)NC(c2n[nH]c(CO)n2)C)CC(NC(c2csnn2)=O)C1(C)C C(CC(F)F)(C(=O)N1C2CCCC1CC2)NC(C1CC12CCCCC2)=O N1(C(C(C)N2CCCC2)=O)CCCN(C(=O)Cc2ccc(Cl)cn2)CC1 CN=c1ccc(C(N2CCC(C(C)NC(c3cnn(C(C)C)n3)=O)C2)=O)c[nH]1 N1(C(C)=O)CCCC(N=c2[nH]c3c(c(=NCC4COCCO4)[nH]2)CSC3)C1 C1(NC(c2ccc(COC)o2)=O)CCOC(C(=O)NCCc2nccc(O)n2)C1 C=C(CNC(C1(C(C)C)CCN(C(=O)CC2CCCC2O)C1)=O)c1ccccc1 C(C)(C1=CCN(C)CC1)NC(C1N(C(COC(C)C)=O)CCOC1)=O C(=O)(CCCC(N)=O)N(CC(CO)(CO)NC(=O)CC1C=CCC1)C Cc1cc(N2CCCC(NC(=O)CCn3cccn3)C2C)ncc1[N+](=O)[O-] N1(C(C(C)NC(CC)(C)C)=O)CCCC1(C)CNC(=O)CCc1ccc(C)cc1 C1(OC)CN(C(=O)CCC2CCCO2)CC1NC(c1c(C(C)=O)cnn1C)=O c1(C(N2CC(CNC(c3n(CCC)ncc3)=O)C(C)C2)=O)cccc(C#N)c1C C(=O)(C1CCc2ccccc21)N1CCC(C)(C)C1CNC(=O)CNS(N)(=O)=O N1(C(CCCC(C)NC(C2(C)CC2(F)F)=O)=O)CCOC2(CCC2)CC1 CC(C)CC(C(=O)N(C)Cc1nnnn1C)N(C(=O)C(C1CC1)C1CC1)C CC1CCN(C(c2cc(C(N)=O)ccn2)=O)CCN1C(=O)CC1CCCC2CC12 C#Cc1cncc(C(N2CC(NC(C3(c4cccs4)CC3)=O)CC(C)C2)=O)c1 N1(C(C(CC2CC=CCC2)NC(=O)OC(C)(C)C)=O)CCc2nccc(Br)c2C1 C(C(C(C)C(C)C)N=Cc1ccn(C)c1)NC(COCCC(C)C)=O CN(Cc1ccncc1)N1CCCC(OCC2CCN(C(=O)OC(C)(C)C)C2)C1 c1(C(=O)NC(C)C(CO)NC(c2[nH]nc3ncccc23)=O)cc2c(s1)COCC2 c1(C(=O)NCC(C)(O)c2cccs2)sccc1CNC(N)=O C=CCC(CNC(=O)CSC1CC1)C(=O)NCc1ccc(OC)nc1 c1(C(C)C)ncc(C(=O)NC2(C)CN(C(C3CC3c3cccs3)=O)C2)n1C C(=O)(C(C)(C)CC1CC1)NC(CC(C)NC(c1ccc(Cl)cn1)=O)C N1(C(C=CCC(C)(C)NC(c2c(C)ccnn2)=O)=O)CCc2c(nnn2C)C1 Cc1cc(C(=O)NCC(C)NC(C2CCC(C(C)C)CC2)=O)[nH]c1C c1(CC(=O)NCCOCCN(C(=O)CSc2ccccc2F)C)cc(Cl)n(C)n1 N1(C(C(C)CC(F)(F)F)=O)CCOC2CCN(C(c3cnn(C)c3)=O)CC12 C(CCC(=O)Nc1ncn(-c2ccccc2)n1)NC(CC)=O C1(C(=O)OC)CC12CC(NC(c1ncoc1CNC(C1CCC1)=O)=O)C2 N1(C(Cc2n(C)cnc2)=O)CC2CC1(C(=O)NCC1CC(C)(O)C1)C2 Cc1nc(NC(=O)CC2CCCN2Cc2cccc3[nH]ncc23)c(C#N)n1C N1(C(c2c(C)n(C)nc2)=O)CC(NC(c2cccc3nccn23)=O)C(N=[N+]=[N-])C1 c1(C(N(CCCNC(C2C(C)(CC)C2)=O)C2CC2)=O)cncc(C(N)=O)c1 C=CCC(C)C(=O)N(C1CCCCC1)CCNC(c1cn(CC(F)F)nc1C)=O C=CCC(CC=C)C(=O)N1CC(CNC(C2CC3(C2)CC2(CC2)C3)=O)C(C)C1 Cc1nc(C)c(CC(=O)NCC(C2CC2)NC(c2cnc(CC(C)C)[nH]2)=O)s1 N(C(=NCCS(=O)(=O)NC1CC1)NC1CC1)CC(c1cccc(C)c1)O N1(C(C(C)N(C(=O)C=CCF)C)=O)CC(O)C(O)C1 C=CCC(C)(C(=O)NCC(C(C)(C)C)NC(C1CN(C)C(=O)N1)=O)N(C)C c1(CCC(=O)NC2CC(N(C(C(C)N(C)C)=O)C)C2)cnc(C2CC2)o1.C1CC1 C(c1cnccn1)=CC(=O)N(CC(C)NC(c1cnc(N(C)C)o1)=O)CCF CCCCCC(=O)NCCN1CCC(NC(=O)CCn2cnccc2=O)CC1 C1(C(=O)NCCC(C(C)C)NC(=O)C(C)(C)c2ccno2)CN2CCC1(C)CC2 C#CCC(CC(=O)NC1CCCCCC1C)NC(C1CC2C(C1)C2(C)C)=O c1(C(=O)NC2CCN(C(C(C)CF)=O)C2)noc2ccc(Cl)cc12 C1(OCC(=O)NC(C)(CNC(=O)C(F)n2cccn2)C2CC2)CCOCC1 N1(C(Cc2nc(C)sc2C)=O)CC(C)N(C(c2cc(C3CC3)[nH]n2)=O)CC1C c1(CNc2scc(-c3c(F)cc(OCC)c(F)c3)c2)cc([N+](=O)[O-])c(C)cc1F N1(C(C)(C)C)CCCC(c2nnnn2C2COC2)(NCCF)C1 C(=O)(C1CCCc2ncccc21)N(C1CN(C(C(=Cc2cccnc2)C)=O)C1)C C1(C(=O)NCC(CC)NC(C2C3C4CCC(C4)C23)=O)CCc2ccc(F)cc2O1 n1(CC(N2CC(CC)C(NC(C3CCOCC3)=O)CC2)=O)ncc2ccccc12 CC1(CNC(=O)CC(F)(F)Br)CCN(C(=O)C=Cc2ccccc2)C1 c1(-c2cn(CC(CNC(=O)Cc3sccc3Br)OC)nn2)nccc(C(=O)O)n1 C1(n2c(-c3cc(F)cc(Br)c3)nc(CCN(C)C)n2)CCOC2(CCCC2)C1 C(C)(C(C(=O)NCCCOCC(C)C)NCC)OC(=O)C(O)CN(C)C c1(COC)nc(=NC(CNC(=O)C(C)SC)C2CCC2)s[nH]1 c1(C(C(=O)NC)N(C(c2ccccc2)C(C)C)C)c(Cl)cnn1C c1(CNC(C2CCN(C(CC(C(=C)C)OCC)=O)C2)=O)cccc(S(=O)(=O)NC)c1 CCCCCCCCCCC(=O)N1CCN(C(C2CCCNS2(=O)=O)=O)C(C)C1 c1(C(N2C(C)CC(CNC(C3CC4C=CC3O4)=O)CC2)=O)c(F)ccc(N)c1F C12(CC(=O)NCc3n(CC)ncc3)CCC1CN(C(C1(O)CCOC1(C)C)=O)C2 c1(C(=O)NCCN(C(=O)CCc2ncnn2C)CCOC)c2c(nn1C)CCC2 N1(C(C(C2CC2)OCC)=O)CCCCC1C1CCCN1c1nnc(COC)s1 c1(CC(N2CCC(NC(CN(CC)CC)=O)C2C)=O)c(C)nn(C(C)C)c1C Cc1cnncc1C(=O)NCC(CO)NC(C1CCC(O)CC1)=O C(=O)(CC(C)(C)C(=O)N1CCCCC(CNC(C2(CC)CCC2)=O)C1)OCC CC1CN(C)CC1C(=O)NCC1(F)CC(NC(=O)CSc2nnnn2C2CC2)C1 C(C(=O)N1CCC(NC(c2ccc(C)cn2)=O)C1C)(C(F)(F)F)OC(C)=O Cc1cc[nH]c(=N)c1C(=O)NCC1CCC(NC(=O)CCS(C)=O)C1 CC(C)C(CNC(C1(CO)COC1)=O)NC(=O)Cc1cncn1C c1(C(N(C)CC2N(C(C3C(C(=O)OC)CCC3)=O)CCC2)=O)cc(CO)oc1C Cc1cnn(C)c1C(=O)N(C)CC1(C)CCCC1NC(C1CC1C1CC1)=O c1(OC)ccc([N+](=O)[O-])cc1CN1CCN(c2ncc3[nH]ncc3n2)C(C#N)C1 N1(C(C(CC#C)(C)C)=O)CCC2(CC1)CC2C(=O)NCC(O)CCC=C C1(CNC(CN2CC(C)(OC)C2)=O)CCCCN(C(c2ncccc2CSC)=O)C1 CC1(C)C(C)(C)C1(F)C(N1CCCC(NC(c2coc(C3CCC3)n2)=O)CC1)=O c1(COC)ccc(OCC(=O)NC2CC(N(C)C(c3ccc(C)cc3)=O)C2)cc1 C1(NC(CC(=C)C)=O)CCN(C2CCN(C(c3cnc(Cl)[nH]3)=O)CC2)CC1 Cc1cc(C)c2c(c1)C(OC(c1occc1CS(=O)(=O)c1ccccc1)=O)CCO2 N1(c2cc(C(C)(C)C)ncn2)CC2CC(NC(c3ccc(CO)c(F)c3)=O)C2C1 c1(C(=O)NC2CN(C(C3C(C)(C)OCCO3)=O)CC(O)C2)onc2c1CCCC2 C1(C(=O)NCCC(C)N(C(=O)Cc2cn[nH]c2)C)CCOCC12CCCC2 CCC(CNC(=O)Cn1cc2ccccc2n1)N=c1[nH]nc(C2CCCC2)s1 CCCC(C(=O)NCC12COC(CNC(C3CCC(F)C3)=O)(C1)C2)NC(N)=O C1(NC(c2c(OCC)oc(C)n2)=O)CC(F)CN(C(=O)Cc2c(C)noc2F)C1 C1(C)(C(=O)NCC(=C)CCNC(C2(OC)CCC2)=O)CCSCC1 C1(NC(C=Cc2ccc(C)o2)=O)CC(C2CCN(C(c3cccc(F)c3)=O)C2)C1 C1(C(=O)NCC=CC(=O)NCCn2c(CC)nnc2)CCCCCCC1 C1(NC(C(C)=CC)=O)CC(CNC(=O)Cc2cc(C)ns2)C1(C)C c1(N2C(C)CC(NC(c3cnc(F)c(F)c3)=O)CC2)ncc([N+](=O)[O-])cc1Br C#Cc1ccc(C(=O)NCCC(CC)(CC)NC(c2cnccc2C)=O)c(C)c1 CC(C)C(F)(F)CC(=O)NCCN(C(C1CCC2(C1)CC2(F)F)=O)C1CC1 c1(C(N2C(C)CCC(NC(=O)C(C)(F)F)C2)=O)cnc2cccnc2c1 Cc1ccc(F)cc1NC(C1(C2CC2)CN(C(=O)COc2ccccc2)C1)=O C1(C(N2CC(C)(C)OCC2CNC(C2(C)COC2)=O)=O)CNC(=O)CC12CCC2 CCC(COC)C(=O)NC(CCN(C(=O)C(F)(F)CO)C)C(C)C N1(C(c2cnn(CCCC)c2C)=O)CC2CCN(C(c3cc(C)c(C)s3)=O)C2C1 N1(CCC(=O)NC(C(C(C)C)=O)c2ccccc2)C(=O)c2ccc(Br)cc2C1=O Cc1nc(C(C)(C)C)ncc1C(N1CCOC(C(F)(F)F)C1C)=O C1(CNC(C(C)NC(=O)CC2CCOC2(C)C)=O)CC12CCOCC2 c1(CCC(N2CC(CCO)(NC(CNC(CC)=O)=O)C2)=O)cnc2n1CCCC2 c1(C(=O)NCC(CNc2ncc(C(=O)OC)cn2)O)c(CC)nc2sc(C)cn12 c1(CC#N)ccc(F)c(-c2csc(C(=O)NC3CCCCC3CO)c2)c1 c1(C(=O)NC(CCN(C(CC(C(C)C)C)=O)C)C(C)C)ccsc1S(N)(=O)=O c1(C(N2CCN(C(CSC(C)C)=O)CC2)=O)cc2n(n1)CCO2 C=CCCCCC(=O)NCC1CC1C(=O)Nc1cnn(C)c1CCC c1(C(N2C(CNC(C(CC)C#N)=O)CC(O)C2)=O)cc(Cl)cc2ccncc12 C1(C(=O)NCCCNC(CCN(C)C)=O)CN(Cc2ccccc2)CC12CCC2 c1(N2CCC(OOC)C2=O)cccc2ccccc12.C12COCC(C)N(C1)C2=O C1(C(=O)NCCC2N(C(c3nnc(C)s3)=O)CCSC2)CN2CCCN1CC2 CC1(C(=O)Nc2nccc(Cl)c2Cl)CCCN(C(=O)CC2COCCO2)C1 N1(C(c2cnc(CNC(C(C3CCC3)OC)=O)nc2)=O)CC2CN(C)CC2(C)C1 c1(NC(C(=O)NCCN2CCCS2(=O)=O)=O)cc(Br)c(F)cc1F c1(C(N2CCOCC2)CNC(C(C2CCCN(C)C2)(C)C)=O)cccc(F)c1F C1(C(N(CC(C)CNC(C2CCC(=O)N2)=O)C)=O)CCC2(CCC2)C1 c1(CNC(CO)Cc2ccccc2Br)cccc(F)c1F Cc1c(F)ccc(C(=O)NCC2CC(C)CCN2C(c2ccsc2)=O)c1N C(=O)(C#CC1CCOC1)N1CC(CC(=O)NC23CC(C2)C3)C1 C(=O)(C1=CN=C2N=CNN2C1)NCC(C)CNC(c1cccnc1C(F)(F)F)=O c1(C(=O)NCC2N(C(CC(=O)NCC)=O)CCN(C)C2)cc2ccc(C)cc2[nH]1 c1(CN(C(C=CC)=O)C)ccccc1CNC(c1ccnn1CCN(C)C)=O c1(C(=O)NCC(C)OCC=C)cc(CNC(=O)C(F)CC2CCC2)nn1C c1(NC(=O)CNC(=O)C(F)(F)F)cccnc1C(=O)NCCN(CC)CC C1(C(=O)NC(C)CCNC(=O)C(C)(C)Oc2ccc(F)cc2)CCCCS1(=O)=O N1(C(Cn2ncc(C)c2)=O)CC(C2CC2C(=O)N(CC(c2nn[nH]n2)C)C)C1 Cc1nn(CC(=O)NC2(C)CC(NC(C3C(F)(F)C34CC4)=O)C2)c(C)c1C CCC(CCOC)C(=O)N1CCOC(CCNC(C2(CO)CC2)=O)C1 C1(NC(C(CC(=C)Cl)NC(=O)CC2CC2C2CC2)=O)CCCC(C2CC2)C1 c1(C(=O)NC2(C)CCN(C(C3(C)CC(C#N)C3)=O)C2)cccc(Cl)c1Cl C(CCCCCN=[N+]=[N-])NC(CC(CC)N(C(CC1ON=C(CC)C1)=O)C)=O C(=O)(C(C)(C)CCOC)NCCN(C(C(F)=CCC)=O)Cc1cccc(Cl)c1 N1(C(C=CCCC)=O)CC(NC(c2scc(C)c2Cl)=O)CC(F)(F)C1 c1(C(N2C(CNC(C(CC)(C)OC)=O)CC(C)(C)C2)=O)ccc(S(C)=O)cc1 n1(CCC)cc(CNC(c2nnnn2C2CCC2)C2CCC2COC)c(C)n1 C1(CNC(c2c(C)cc(C(=O)OC)o2)=O)CN(C(C2CCOCC2)=O)CCCO1 c1(C(=O)NCC2C(CNC(C(CC)(C)O)=O)C2)cc2n[nH]cc2cc1C c1(CNC2CC(NC(c3cc[nH]n3)=O)C2)ccc(I)cc1O C1(C(N2C(CNC(C3(OC)CC3)=O)CC3CC32)=O)CCc2nccn2C1 C1(F)(CNC(Cn2ncc(C)c2)=O)CCN(C(c2ccc(Br)cc2)=O)CC1 Cc1ccc2[nH]nc(C(=O)NC3CCC4CCN(C(C5CCCS5)=O)C34)c2c1 C1(NC2CC(c3ccc(F)cc3)C2)CCCCCC12CCCC2 c1(C(C(=O)NC(CC)C)N(CCCCCO)C)cn(-c2ccc(Cl)cc2)nc1C C1(c2cc(CC)no2)CCCCN1C(c1nnc(-c2cccc(Cl)c2)o1)=O C1(C(N(C2CCCN(C(c3c(C)nc(CC)o3)=O)C2)C)=O)CCC2CCC1O2 c1(CNS(=O)(=O)NC2CC(c3ccc(Cl)cc3)C2)cccc(Br)c1 c1(CN(C(C(=O)NC(C)CN(C)CC2CCCCO2)=O)CCO)ccc(Cl)cc1 CN1CCN(C(=O)CSCCNC(c2cn(C)c(=O)cn2)=O)CC1=O C1(CC(=O)N(CCCN(C)Cc2sccc2Cl)C)CC(C)(C)CO1 C1(CC)CCCCN1C(=O)C(C)N(CCCNC(c1cc(C(N)=O)co1)=O)C C1(N(C)C(c2cc(Cl)nn2C)=O)CCCCC1NC(c1csc(C2CC2)n1)=O c1(C(C)C)cccc(C(N2CCC(NC(=O)C(c3cccc(F)c3)O)CC2)=O)c1 c1(C(N2C(CNC(C(COC)(C)OC)=O)CC2)=O)ccccc1P(C)(C)=O N1(C(c2onc(C)n2)=O)CCCCC1CNC(C1CC2CC2C1)=O N1(C(c2cc(C(C)(C)C)on2)=O)CCCCC1C(N1C2CCC1CC2)=O c1(C(N2CC(O)(CCNC(C3C(C)CC(=O)NC3)=O)C2)=O)cc(F)cc(Cl)c1N N1(C(C(c2ccn(C)n2)C)=O)CCC1(C)CC(=O)NCCCOC(=N)O c1(N2C(C(=O)OCc3ccnc(F)c3F)CCC2)ncnc2ccccc12 C(=O)(CC1=CCCC1)NCCN(C(=O)C=Cc1cnccn1)C(C)C c1(COCCOCCOCC)cscc1S(=O)(=O)c1ccc(C)cc1.C1C(=O)O1 C(=O)(C(CC(C)C)NC(c1ncn(C)n1)=O)NCC(CSC)OC C(c1ccc2occc2c1)=CC(=O)NC1(CNC(C(COCC)C)=O)CCOC1 C(C(=O)NC12CC(C(=O)Nc3cc(Br)c(C)s3)(C1)C2)(C(C)C)OC N1(C(c2n(C(C)C)nnc2)=O)CCn2ncc(CNC(C3CCCOC3)=O)c2C1 CCCCC(C)(C)NC(=O)C(Cn1cncn1)NC(=O)C(C)C(=O)OC C1(C(=O)OC)(C(=O)O)CC(NC(=O)C(n2cc(-c3cnc(NC)s3)nn2)C)C1 CC(CC(N)=O)C(=O)NC1COCCN(C(c2ccc(SC(F)(F)F)cc2)=O)C1 C(=O)(C1=C(C#N)CCC1)N1C2CC(CNC(Cc3nc(C(C)C)sc3)=O)C1CC2 Cc1cc(C(=O)N(C)CCNC(=O)CC2C=NN(C)C2=O)ccc1C#N c1(C(=O)NCC2CCN(C(C(F)=C(C)C)=O)CC2C)cncc2c(O)nccc12 C(=O)(C(F)(F)CNC(=O)Nc1ccc(C(C)(C)C)cn1)OCC N1(C(C2C(C)(C)C2)=O)CCC2C(NC(C3(C)C=CCCC3)=O)C2C1 Cc1nc[nH]c(=NCC(C2CCCC2)NC(=O)C=CC2CC2)c1C#N C=Cc1cncc(C(=O)NC(C2CCCCC2)CNC(=O)CN(C)S(N)(=O)=O)c1 C(=O)(C#CC(C)C)N.C1(C)(OC2(CC=CC(=O)NCC)CCC2)CNC1 c1(N2CC=CC(NC(CC3(COC)CCCC3)=O)C2)ccc([N+](=O)[O-])cc1 C1(CNC(CCC2(NC(CN(C3CC3)CC)=O)CCC2)=O)CCN(C)CC1 C1(NC(C(C(=O)OCC)F)=O)CC2COCC(C1)C2NC(=O)CCC1CC1 C1(O)(CNC(c2ccc(NC)cc2)=O)CCCN(C(c2scc(C)c2Cl)=O)C1 N1(C(C2CCC(=O)NC2)=O)CCC2(CCN(C(C3CCCCCC3)=O)CC2)C1 c1(C(=O)NCC(CN(C(c2cncc(SC)c2)=O)C)O)cc(C(N)=O)ccc1C C(CCF)(C(=O)N1CC(C(=O)NC)C1)NC(Cc1onc(CC)n1)=O C(CN=c1c(C)c[nH]cc1[N+](=O)[O-])C1CCC(NC(C2=C(C)OCCS2)=O)C1 N1(C(C(C)C)=O)CCCC(C2CCCCN2C(c2ccnc(C3CC3)c2)=O)C1 N1(C(C2(COCC)CC2)=O)CC2CC1CN2C(=O)Cc1cccc(OCC)c1F C1(NC(CCSC)=O)CN(C(C2CC3C(C2)C3(C)C)=O)CC12CC2 c1(CC)cccc(C(=O)NCCCN2CCN(C(C3CCCN(C)C3)=O)CC2)c1 C1(CC(N2C(CN(C(c3nc(Cl)c(CC)[nH]3)=O)CC)CCC2)=O)CCCCN1C C1(C(N2CCN(C(N)=O)CC2)=O)CC2(CCC2)CN1C(=O)CCN1CCCCC1 c1(C(=O)OC)nc(C(=O)NC2CCC(CNC(C3CC(OC)C3)=O)C2)cs1 C(CC(=O)NCC1C=CCN1C(c1ccc(O)nn1)=O)(C(F)(F)F)OC N1(C(C2C3(CCN(C(c4cccc(CO)n4)=O)C3)C2)=O)CC2CCOC(=O)C2C1 N1(C(C2CC(NC(=O)C(F)(F)C3CC3)C(O)C2)=O)CCc2ccsc2C1 C1(NC(CCNC(=O)NC)=O)CC(CNC(=O)C=CC(C)(C)C)C12CCC2 C(=O)(C#CC1CCC1)NCC(CCCC)NC(=O)CCOC1CCC1 C1(C2CC2)(CC(=O)N(CCNC(C2(NC(CC)=O)CC2)=O)C)CC1 C(=O)(C1(C)CCOc2ccccc21)N1CC2C(NC(C3(OC)CCSC3)=O)C2C1 C(=O)(C=C(Cl)Cl)NCCN(C(=O)C(c1ccccc1)n1cccn1)C(C)C c1(C(N2CC(C(=O)NCc3ccc(C)c(C)c3)SCC2)=O)cc(Cl)c(C)c(Cl)c1 c1(CN2C(C(=O)Nc3c(CC)ccc(Br)n3)CC2)cc(OC)c(OC)cc1OC N1(C(=O)Nc2ccc(Br)nc2F)CCCC12CCOC2 CC1CN(C(C2CC3(C2)CC(O)C3)=O)CCN(C(=O)C(c2ccn(C)n2)C)C1 C1(NC(c2onc3ccccc23)=O)CC12CCN(c1nccc(Br)n1)CC2 c1(C(N2C(C(N3CC(C)(CCO)C3)=O)C=CC2)=O)ccncc1F CC(C)C(C(=O)N1CCC(C)(CCNC(=O)COC2(C)CCC2)C1)NC(N)=O Cc1nnc2n1C(C(=O)NCCN(C)C(C1(c3ccccc3)CC1(C)C)=O)CC2 Cc1ccc(OC(F)F)cc1C(=O)NCCCN(C(=O)C=Cc1ccoc1)CC CCN=c1[nH]c(C(=O)N(C2CCC(CNC(=O)C(F)=C(C)C)CC2)C)cs1 C(=O)(CCC(=O)NCCCC1CCN(C(=O)COCC2CC2)CC1)N(C(C)C)C C(C1CCCCCC1)=CC(=O)N(C1CCN(C(C2CCN(C)S2(=O)=O)=O)C1)CC n1(CC(=O)NC(CCNC(C=CC(CC)=CC)=O)C)cnc([N+](=O)[O-])c1 c1(-c2nc(C)sc2)cc(CNC(C2CC2c2cn(CC(=O)O)nn2)=O)n(C)c1 C1(C(N(C)CC2CCSCC2)=O)CC12CC(NC(c1ccncn1)=O)C2 N1(CCCN(C(=O)NCCCCCCF)CC)CCN2CCCC2C1 CC(C(C)(C(=O)O)C(=O)O)NC(C1(C)CCC(F)(F)C1)=O C1(CC)(CNC(C2OCCC2CNC(=O)CC2CNC(=O)O2)=O)CCC(=O)N1 N1(C(COC(CC)(C)C)=O)CCC2(CNC(=O)C(C)c3cccs3)CCCCC12 C12(CNC(c3c(CCC)nns3)=O)CCC(CC1NC(=O)Cc1nonc1C)C2 c1(C(N2CCC(NC(C(CC#C)(C)C)=O)CC2C)=O)occ2c1CCOC2 c1(C(N2CCC3(CN(C(C4(C)CC(=C)C4)=O)C3)C2)=O)cc(=O)c2ccccc2o1 CCC(O)CC(=O)NCCn1cnc(C(=O)N(C2CC(SC)C2)C)c1 C(CCCCC(=O)NC1CC2(C1)CC2NC(c1cc(C2CC2)n(C)n1)=O)=CC c1(C(C)C)ncc(Br)c(=NC2CC(NC(c3cccc(F)n3)=O)C2(C)C)[nH]1 CCCC(CCCO)C(=O)NCC1CN(C)CCN1C(=O)CC(C)(C)CCOC C12(CNC(=O)CSC(F)(F)F)CC(NC(=O)Cc3ccn(C(F)F)n3)(C1)C2 CCCCCCC(CC)C(=O)NCC1(C(C)NC(c2cc[nH]c2)=O)CC1 Cc1cc(=NCCc2nnc3cccnn23)[nH]c(=NCc2cc(Cl)c(Cl)n2C)[nH]1 C1(C(=O)NC2CCN(C(C(C(CC)O)C)=O)C2C2CC2)C2CCC1(C)C2(C)C CCC(C)(C)CC(=O)NC1CC2CC(NC(=O)CC3(C)CC3)C2C1 N1(CCCCOC(=N)O)CCN(C(=O)NCCCc2cncnc2O)CC1 CC(CC(=O)NC12CCN(C(C3CC(OC4CC4)C3)=O)CCC1C2)CC(C)(C)C C(=O)(C(F)F)N(CCCOCCN(C(C)=O)C)C.C=CCSCC1CC1 c1(OC)cc(CN(C=O)Cc2nc(-c3ccccc3I)cs2)c(F)cc1Cl C(CC(C)(C)CC(=O)N(CC(C)NC(c1ccc(COC)cc1)=O)C)OC c1(OC)cc(C(=O)NC2CC(N(C)C(c3occc3F)=O)C2)ccc1C(F)F c1(NC2CCN(C(C3CCCCC34CCC4)=O)C2)ncnc2sc([N+](=O)[O-])cc12 c1(C(C)C)nc(CC(=O)NCCCC2CCC2CNC(=O)CCc2cnc(O)[nH]2)cs1 N1(C(CCOC(C)C)=O)CCC2CC(NC(c3c[nH]c(=O)cn3)=O)CCC2C1 N1(C(c2ccn(CC)n2)=O)CCCCC(C(=O)NCC2NC(=O)NC2=O)C1 Cc1cccc(-n2c(CC#N)nnc2SCCc2scnc2C)c1 C1(CCC)CN(C(C2CCN(C3CC3)C2=O)=O)CCN1C(=O)C1CC1 c1(C(=O)NCCC(=O)N(CCCNC(c2n[nH]cc2Cl)=O)CC)ccccc1Cl C1(N(C(C(C)N(C(=O)C(O)CC2CCCC2)C2CC2)=O)C)CCCC1(F)F C(C)(C(C)C(=O)NOCC(C)(C)O)NC(C(C)CC#N)=O CCCC(C(=O)N(C1CCN(C(c2cc(C)nc(O)n2)=O)C1)C)C(C)C c1(C(=O)NC(C(CCC)C)C)n[nH]c2c1CN(C(=O)CCC1CC1C)C2 CC(C)(CF)C(=O)N1CC2C(C(=O)NCCC#CCO)C2C1 C1(C(=O)NCC23CN(C(c4c(C)ncs4)=O)C(CC2)C3)CCc2cnn(C)c2C1 C1(CNC(CC=C)=O)CN(C(=O)C(C)Oc2ccc(C)cc2)C(C)(C)C1 CC1CCCN1CC(=O)NCC1CC(NC(=O)C(C)(C)Oc2ccccc2)C1 N1(C(COC(CC)C)=O)CC2(C(=O)NC3CC=CCC3)CCC1CC2 Cc1cc2c(CC(N3C(CNC(=O)C(O)CF)CC4CC34)=O)csc2s1 c1(C(=O)NCCCC(=O)NCC(CC)OC(C)=O)nn(C)c(C2CC2)c1C N1(C(CCc2cn(C)nc2)C(=O)NCc2cccs2)CCC2(CCC(O)C2)C1 c1(C2C(Nc3[nH]nc(CCSC)n3)C2)cc(OC(F)F)ccc1F O=C1NCCCCC1C(N1CCCCC1CC(N1CCC(n2ccnn2)C1)=O)=O C(C(=O)NC1CCN(C(=O)COc2ccccc2)CC1O)(C(C)(C)C)N(C)C C1(CC=C(C)C)CCCN(c2ccnc(NC3CCN(C(=O)C(C)C)CC3)n2)CC1 c1(OC)ccc(C(C)NC(c2cc(C)ccc2F)=O)c(Cl)n1 c1(C(N2CCC(NC(C(C)c3cccs3)=O)C(F)C2)=O)onc2c1CCCC2 c1(CC(=O)NC2(CNC(CC3CCC(=O)N3)=O)CCCC2)cnc2cccnn12 C1(NC(C2(COC)CC(=O)C2)=O)C2CC3C1C3C2C(=O)NC(C)CC1CC1 CC(CC(=O)c1c[nH]cn1)(C(=O)O)c1ccccc1 CCC(CNC(=O)CNC(c1ccccc1)=O)(CC)Sc1nn[nH]n1 N1(C(c2cc(C)sn2)=O)C2CCC1CC(C(=O)NCC13CCCN(CC1)C3)C2 C1(NC(CCc2c(C)nn(C)c2)=O)CN(C(=O)C(C#N)C2CC2)CCC1CO CC(CS(C)(=O)=O)C(=O)N(C1CCN(C(c2ccc(S(N)(=O)=O)o2)=O)C1)C c1(C(=O)NC(CCC)C(=O)OC)cn2c(n1)CN(C(c1ccc(C)cc1)=O)CC2 C(=O)(C1=CCC(F)(F)CC1)N1CC(N(C)C(c2ccnc3c2CCC3)=O)C(F)C1 C1(NC(NCC2(OC)CCCC2)=NCc2ccccc2)CC(C)(C)CC(C)(C)C1 c1(C(=O)NC(CC)CN(C(=O)C(O)C(C)C)C)nc2n(c1Br)CCC2 C1(NC(c2c(F)ccc(C)c2)=O)CN(C(c2ccncc2O)=O)CC(F)(F)C1 N1(C(c2c(CC)noc2)=O)CCCC(N(C(=O)CSc2c(C)n[nH]c2C)CC)C1 N1(C(CC(=C=C)C)=O)CCC(n2cc(COC(=N)O)nn2)C(O)C1 C1(CC(C(=O)NCCOC)N(C)Cc2ccc(C)s2)CCC(C)(C)O1 N1(C(C(C)SC(C)C)=O)CCC(C)(C)C1CNC(=O)C=CC1CCCC1 c1(C(N2CCN(C(C3C(=O)OCC3)=O)C(CF)C2)=O)cn2cnnc2cn1 C1(NC(CC2CC(SC)C2)=O)CCN(C(=O)Cn2cc(C#N)cn2)CC1F c1(C(N2C(C)CC(NC(=O)CC3CC=CC3)C2)=O)cccc2nc(Cl)cn12 C(C(C)(C)CNC(c1n[nH]cc1Cl)=O)N(C(C(C)NC(=O)OC(C)(C)C)=O)C c1(C(N2CC(O)(C(C)NC(CCC=C(C)C)=O)C2)=O)ncnc(C)c1C N1(C(COc2cc(C)on2)=O)CCC(C)CC1CNC(C1CCCC2(CC2)C1)=O N1(C(=O)NC2CCOCC2)CC2CC1CC2CF C1(C(=O)NC2C=CCN(C(=O)CC(C)n3cccn3)C2)(COC)CCC(=O)N1 c1(NC(=O)CN2CCCCC2)nc2c(cc1Cl)C(=O)OC2.N12CCC1CC2=O C1(CC(=O)N2CCCC2)CC2CC2C1.C1(C)C(=O)N1C.CCC(=O)OC C1(C(CC)(C)C)CCC(C(=O)NCC(O)CCNC(=O)CCC)CC1 c1(-c2ccc(C(=O)Nc3cccc(C(=O)OC)c3)c(F)c2)cnc2[nH]ccnc1-2 C1(N=[N+]=[N-])(C(=O)NCCc2cc(C)no2)CCN(C(=O)CC2(O)CCCCC2)C1 N1(C(CN2CCC(C)C2)=O)CCCCC(NC(C2(O)CC2)=O)C1 Cc1ccnnc1C(=O)NC1CC1CNC(c1nc(C)n(-c2ccccc2)n1)=O C1(NC(c2ccnnc2)=O)CN(C(C2CC23CC3)=O)CC1C(F)F c1(C(=O)NCCC(C)NC(CC=C=C)=O)cnn2ccncc12 C(=O)(CCCC(=O)N1C2CCC1C(CNC(c1cnsc1)=O)C2)NCC c1(OCC)cc(C(N2CC(NC(C3NC(=O)C4CCC34)=O)C2)=O)cc(Cl)c1O C(=O)(CC(C)C(F)(F)F)NCc1nc(C)c(C(=O)NC(C)(CO)C(C)C)o1 Cc1cc2cc(CNC(=O)C(=O)NC(C)COC(C)(C)C)ccc2[nH]1 C(=O)(C1CCCc2ccnn21)NCC1N(C(c2c(CC)nc(C)n2C)=O)CC1 CCC(C(=O)NCC1(N(C(=O)C(CSSC)NC(C)=O)C)CC=CC1)N(C)C c1(C(=O)NC(C(C)C)CNC(=O)C(C)n2cnnn2)coc2cc(F)ccc12 Cc1nnc2n1CC(CN1CC(NC(C3CCCCS3)=O)C1)CC2 N1(C(C2(C#C)CCCC2)=O)CC(NC(=O)C(C)SC(C)C)C2(CCC2)C1 C12(C(C)=O)CC(C(N3CC(C(C)NC(c4cc(CC(C)C)c[nH]4)=O)C3)=O)(C1)C2 N1(CC)CCC=C(c2cn3cc(C(N4CCN(CC(F)F)CC4)=O)ccc3n2)C1 C(=O)(C#CC1CCCCC1)N(C1CCN(C(C2(C)CCNC2=O)=O)CC1)CCC c1(C(=O)NC(C(C)NC(C=CC(C)C)=O)C(C)C)nccc2c(Cl)cccc12 c1(OC)ccc(C(=O)NC2CN(C(c3ccc(C4CC4)cc3)=O)C2)cc1C CC(C)C(C(=O)N1CC(O)C(N=[N+]=[N-])C1)C(C)NC(c1ccnn1C)=O N1(CCCCNC(C(COC)O)=O)CCCN(C(c2cc(F)ccc2O)=O)CC1 n1(CCCSCC)nnnc1C(c1ncoc1C)NC(c1nnc(C)o1)CSC N1(C(CCC(C)(C)NC(=O)Cn2cc(C#N)cn2)=O)CCn2cncc2C1 CCCCC(C)C(=O)NCC(O)CNC(c1cscc1CC)=O N1(C(C2(C)CCCCC2)=O)CC2CCC1C2NC(=O)CCC1CCC(=O)N1 c1(C(c2nnnn2C2CC2)NC(CC=C)C2CC2)ccc2c(c1)CCCO2 Cc1[nH]c(-c2ccccc2)c(C)c1C(=O)N(C)CCN(C)C(C1COCCO1)=O c1(C(N2CCCN(C(C3CCCO3)=O)CC2)C(=O)NCC)c2c(nn1C)CCC2 CC1(C(N2CCC(OCCNC(c3ccc(N)c(N)n3)=O)C2)=O)CCC(F)(F)C1 C1(C(=O)NCCN2CCCNC2=O)C2CCCC2CN1C(=O)COCCF C1(CC=C)(C(=O)NCC(C)(O)COC)CCCN1C(=O)CS(=O)(=O)NC N1(C(=O)OCCCc2ccc(C(F)(F)F)cc2)CCC(C(O)C(F)(F)F)CC1 c1(CC)nc(C(=O)NC(C2CCCN2C(c2cc(C3CC3)no2)=O)(C)C)cs1 N1(CC(C(CC)C)NC(=O)OC(C)(C)C)CCC12CC(CNC(C)=O)C2 C(=O)(C(C)(C1CC1)N(C)C(c1c[nH]nc1Cl)=O)NCC(C1CC1)SC N(C(=NCCC1CC(C)(C)CO1)N1CCC2CCCCC2C1)CC(C)C C(CCCCCC(=O)NCC1CC(C)N(C(c2cncc(O)c2Cl)=O)C1)SC N1(C(CCC(=O)c2ccncc2)=O)CCN(C(C2CCCCO2)=O)C2(CCC2)C1 c1(C(=O)NCC(C)(CO)NC(C(CCSC)N(C)C)=O)c(C)nc2sc(C)cn12 C(C)(C)(CCCC(=O)NCC(N1CCOCC1)C)NC(c1c(C)cc(F)cc1)=O c1(C(=O)NCC(COC)NC(=O)CCc2csc(C)n2)n[nH]c(C)c1Cl C#CC1(C(=O)NC(C)C(C)SC)CCN(C(C2CCCN2C2CC2)=O)CC1 N(C(=NCCCCC1(C)OCCO1)NCc1ccccc1)CCCCCC(C)=O N1(C(c2n(CC)ccc2)=O)CCCCC(NC(=O)COCc2nccn2C)C1 Cc1ncncc1C(N1CC2C(CNC(C3(C)CC(C)(C)C3)=O)C2C1)=O N1(C(C(C)Oc2ccccn2)=O)C2CCC1(CNC(=O)C(C)n1ccnc1)CC2 C1(CNC(=O)NC2C=C(C)CCC2)CCCCC1P(C)(C)=O C1(CC)(CNC(c2nnnn2CCSC)(C2CC(C)C2)C)CCOCC1 N1(C(CC2N(C(c3ccc(C#C)nc3)=O)CC(O)C2)=O)CCCC(C2CC2)CC1 Cc1cc2ncc(C(N3CC(NC(=O)CC4=CCCC4)CCC(O)C3)=O)cc2[nH]1 CCCC(O)C(=O)N1CC2CC2(CNC(c2cc(C3CC3)ccn2)=O)C1 C1(NC(C2(NC(c3c(O)cccc3F)=O)C(C)CCC2)=O)CC2(CCCCC2)C1 N1(C(c2c(C)cc(Cl)c(Br)c2)=O)CCOC2CN(C(c3cc[nH]n3)=O)CC12 CC1(C(=O)N2CCC3(C2)CN(C(C2CCCO2)=O)CCO3)CCc2ccccc21 CCCCC(C(=O)NCC12CC1CN(C(c1ccc(=O)oc1)=O)C2)C(C)C c1(C(CNC(C2(C=C)CC2)=O)NC(=O)C(CC)n2cncn2)ccccc1OC N1(C(CC(CNC(c2ncc(F)cn2)=O)C2CCC2)=O)CC2CC(CO)C(C2)C1 Cc1ncnc(C)c1CC(=O)NCC1(F)CC(NC(c2cc(C(N)=O)cs2)=O)C1 N1(C(C=Cc2ccc(C(=O)OC)o2)=O)CCC2CN(C(=O)C3=C(C)OCC3)CC12 Cc1nc(C(=O)NC(C)CN(C)C(C2CC3CC3C2)=O)c(-c2ccc(F)cc2)s1 C12(C(=O)NC(c3ccccc3Cl)C(C)C)CC(C1)C(C(F)(F)F)O2 c1(C(=O)OC)cc(F)cc(S(=O)(=O)NC(C)(C)C(=O)NCC(N)=O)c1F Cc1ccnnc1C(N1CC(O)(CCNC(C2(C)CCCC2O)=O)C1)=O c1(NC(C2(C(=O)OCC)CCCC2)=O)ccc(NC(C2CC3CC3C2)=O)cc1C c1(C(c2nnnn2C2CCOC2)NCC2=C(C)CCC2)cn2cc(C)ccc2n1 C1(NC(C)(CCI)c2nnnn2CCCC2CC2)CCC2(CC1)CS(=O)(=O)C2 N1(c2nnc(C)o2)CCC(NC(C2(C#N)CC(=O)C2)=O)C(C)C1 c1(C(=O)NCCC(C)NC(=O)CCC2CCN(C)C2)c[nH]cc(F)c1=O c1(C(C(N2CC3C(NC(C4CCCC4(F)F)=O)(C3)C2)=O)(F)F)cccc(F)c1F Cc1cc(C)c2nc(N(C3CCNC3)CCO)sc2c1.C(=O)C1=CCCCC1 N1(C(C)=O)CCCC(c2cccnc2)C1.C1C(C)(Cn2cccn2)N1C(=O)C(F)F C1(CNC(C2C(OCC)C2)=O)(NC(=O)C(C)C(C)(F)F)CCCCC1C O=S1(=O)CC2CC(Nc3ncc(Cl)cn3)CC2C1 N1(C(C2(CC=C)COC2)=O)CCC2CCN(C(c3cnn4c3CCC4)=O)C2C1 c1(OC)ccc2ccc(C(=O)NC3(c4cccc(Cl)c4)CCC3)cc2c1 CCCC(C)(CC)C(=O)NC1CC(CNC(c2ncc(F)cc2F)=O)C1 CC12CCN(CC1)CC2C(N1CCC(NC(c2ccsc2)=O)CC1)=O C1(C(=O)NC(CNC(c2ccn(C(C)C)n2)=O)C(C)(C)C)SC2C=CC1CC2 C(=O)(C#CC(C)(C)O)N(C)CC1CCCC1NC(=O)Cc1cccc(Cl)c1 c1(C(=O)NC(C(C(C)C)C)CNC(=O)C=C2CCC2)cc2c(s1)CCCNC2=O C12(C(=O)NCC(=O)OC)C(NC(c3cc[nH]c3C)=O)C3CC1C2C3 N1(C(C(c2ccc(Cl)s2)C)=O)CC2(CNC(c3ccccn3)=O)CC(F)(C1)C2 C(=O)(C#CC1(C)CCCO1)NC1CN(C(Cc2cccc(SCC)c2)=O)CC1C CCC(C)(C)CCS(=O)(=O)N(c1ccc(OC(C)C)cc1)CC(C)C c1(CNC(=O)NCC(CCN(C)C)(C)O)ccccc1[N+](=O)[O-] C(CC(C)C)(C(=O)NCC1CC12CC2(F)F)NC(c1n(CC)ncc1C)=O c1(CNC(CCC)CCC)ccc(SC)cc1OC Cc1ccccc1C(C)NC1CC(NC(N2CCC2)=O)C1 N1(C(C(CSC)O)=O)CCC(NC(c2nc(C)n(-c3ccccc3)n2)=O)CC1C CC(C)CCC(F)C(=O)NCC1(C)COCCN(C(=O)Cc2nc[nH]n2)C1 O=C(C(CCc1ccc(F)cc1)N1CCCCC1CCC(F)(F)F)NCC1CC1 CC(Cc1cnn(C)c1)C(=O)NCCCN(C(=O)CCC1CCOC1)CCO CC1C2CCCCC2CN1C(=O)C(Cc1cn[nH]c1)NC(=O)Cc1cscn1 c1(-n2ccc(C(N(C(CNC(C3(C#N)CCC3)=O)C3CC3)C)=O)n2)ccc(F)cc1 C#CCC(C)(C(=O)N1CC(C)(C)C1C(=O)OC)NC(=O)CC1C=CCC1 c1(C(c2cncs2)NC2(C(F)(F)F)CC2)ccoc1C(F)(F)F C(C(=O)NCCCF)(C1=NOC2COCC12)N(C1C(C)C1)C.c1(C=O)nnnn1C N1(C(CC)C(=O)OC)CC2CC2(NC(=O)N(CCCO)Cc2ccccc2)C1 c1(C(=O)NCCCN(C(c2c(C(C)C)con2)=O)C)cc(F)c2ccccc2c1 C(CCCCCCCO)=CC(=O)NC1C(C)CN(C(=O)Cn2nnc(=O)[nH]2)C1 C1(CC#C)(C(=O)NC(CN(C)C)C(=O)NC(CC)C=O)CCCO1.OC C1(NC(C2(CNC(C(CSC)O)=O)CCCO2)=O)CC2CCCCCC12 c1(NC(C=CC(=O)NCCN(C(c2ncoc2C)=O)CC)=O)cccc(C)c1 c1(C(=O)NCC#CC(=O)N(C)CC2CCSC2)cccc2nccn12 C(CC(CC)C(=O)N1CCOCC1CNC(=O)CCOc1cccnc1)=CC C1(C(=O)NC2CN(C(CN(C3CC3)CC)=O)CC(F)C2)CCc2nn[nH]c2C1 C(=O)(C(C#N)C(C)(C)C)NC(CC#C)CC(=O)NC1(C(N)=O)CCOC1 C=CCC(C(=O)NCC1(CNC(=O)CC(C)c2ccco2)CC1)NC(C)=O C(=O)(C1CCc2nccn21)N1C(C(=O)NC(c2cnc[nH]2)C)CCCC1 c1(C(=O)NC2(CF)CCN(C(c3c(SC)ccs3)=O)C2)cc(C)nnc1O c1(N2CCCC(C)(CNC(C3CCN(C4CC4)CC3)=O)C2)ncnc2[nH]cnc12 C1(NC(c2cc[nH]n2)=O)CC12CCN(C(=O)CCCc1ccncc1)CC2 N1(C(C(C)C#N)=O)CCC(C)C(NC(c2ccc(F)c(C(F)F)c2)=O)C1 N1(C(c2n(C=C)nnc2)=O)CCC(NC(c2cnc(C(F)(F)F)cn2)=O)CC1C N1(C(CC)C(=O)OC)CCN(Cc2cccc(C(C)C)n2)CC1.C12CCN1C2 C(=O)(C#CC1CCOC1)N(C1CN(C(c2cc3n(c2)CCCC3)=O)CC12CC2)C O=C(CCC(=O)N1CCOCC1)NCC(O)CCNC(=O)C1CC1 C(=O)(C1CC(O)c2ccccc21)NC(CC)CNC(c1cc(Cl)ncc1OC)=O c1(CN2C(CCC(=O)NCc3nccc(OC)c3)CCC2)c(F)ccc(F)c1F c1(-c2nc(C(CCC)OCc3ccccn3)n(CCOC)n2)ccc(Cl)cc1O c1(-n2cc(CN(C(CC)CC)C)nn2)ccc(OC)cc1 c1(C(=O)NC(C2(CNC(C(F)OC)=O)CC2)C)sc2nc(C)cc(C)c2c1C CC(C)CCC(F)C(=O)N1CCCC1C(=O)NC(c1nc[nH]n1)C1CC1 CC(C)C(CC(=O)N1CCOC(C(C)NC(c2ccncc2F)=O)C1)C(C)C C1(C(=O)Nc2cccc(CNC(CC3CC(C)C3)=O)c2)CC(C)(C)OC1(C)C c1(OC)ccc(CNC(C2(F)CN(C(=O)CC3CC(=O)C3)C2)=O)cc1C(F)(F)F Cn1cnc2c(NC3C4CCCC34)nc(N3CC4CCC(C3)N4C)nc12 c1(C(N(C2CCCN(C(=O)Cc3c[nH]ccc3=O)C2)C)=O)ccc2scnc2c1 N1(C(C(C)NS(CCC)(=O)=O)=O)CCN(C(c2n[nH]c(CC)n2)=O)C(C(F)F)C1 S(=O)(=O)(c1cc(Br)c(Br)s1)N1C2C(C(=O)Nc3ccnc(Br)c3F)C(C2)C1 C12(CNC(c3n(CCOC)ncc3)=O)CN(C(=O)C=C3CCCC3)CC1CCO2 CC(C)C(O)CC(=O)NC1CN(C(c2cn(C)nc2Cl)=O)CC1c1nccn1C N1(C(CCOC(C)=O)=O)CCCCCC1CNC(C1C2CCN1CC2)=O c1(CC(NS(N)(=O)=O)C)cccc(OCC(N2CCCC2NC(=O)C(O)CF)=O)c1 N1(C(CCSC)=O)CCC2(CCCN(C(=O)C(C)n3cncn3)C2)C1 c1(C(=O)NCC2N(C(C(C(=O)OC)C)=O)CCCCC2)nn(C)c2c1CCCC2 c1(C(=O)NCC2N(C(Cc3cn(C)nc3Cl)=O)CC2)cc(O)nc2c1CCCN2 C=CCC(CO)NC(=O)C(C)(C1CC1)N(C(=O)C(C)=C1CC1)C N1(C(c2csnn2)=O)CCN(C(=O)CCn2cccc2)C(c2cn[nH]c2)C1 c1(OC)cc(Br)c(OC)c(C=NNC(=O)NCc2ccc(F)cc2)c1 C(=O)(C(O)C1=CCCCC1)N1C(C(N2CCC(C#N)(F)C2)=O)CC1 C=C=C(C)CC(=O)NC(C1(O)CN(C(c2cnn(CC(F)(F)F)c2)=O)C1)C N1(C(c2c(C)onc2)=O)CC2CC2(NC(=O)C(C)C2(O)CCC2)C1 c1(SC)cc(C(=O)NCC(C)(C2CC2)NC(c2coc(C)n2)=O)co1 c1(CC)cc(F)ccc1C(N1CCC(NC(=O)CC2CC=CCN2C)C1CC)=O c1(C(=O)NC2C(NC(C3CCN(CC(C)C)C3)=O)CCC2)cnn2cnnc2c1 N1(C(CCCOCC=C)=O)CCC(CO)(CNC(=O)C(C)OCC(F)(F)F)C1 Cc1nncn1NC(=O)C1CC(C)CN(C(C2(F)CCCCCC2)=O)C1 C1(C(=O)NCc2ccccc2)CN(C(=O)C(O)C2CCC2)C2(CCC2)C1 C(=O)(C1=NOC(C)(C)C1)NCC(CNc1snc(C)c1C#N)O c1(C(=O)NCC2CN(C(CCCN(C(C)=O)C)=O)C(C)C2)cc(Cl)ncc1O C12(NC(COCCC)=O)CCN(C(c3cnn(C(F)(F)F)c3)=O)CC1C2 c1(C(C(=O)NCCC#N)N(CCC(C)C#N)c2ccccc2)nn(C)nc1Br c1(NC(c2cc(C3CCCN3)[nH]n2)=O)nncn1C1CC1 CCC(C(=O)NCCOC1CN(C(C2(C3CCCCC3)CC2)=O)C1)C(F)(F)F c1(CC(=O)NCCC(C)NC(C2(O)CC2(C)C)=O)nccc2ccccc12 c1(C(N2CC(CNC(CCC3N(C)CCC3)=O)OCC2)=O)cccc(=O)n1O C(=O)(C1=NOC2COCC12)NC(CCOC)CNC(C12CCC(CC1)C2(C)C)=O CCCCC(C)CCC(=O)NC1CN(C(=O)C=Cc2nccs2)CCC1O c1(OC(F)F)cc2nn1C2.C12C=CCCC1N2.c1(C)ccccc1.CO N1(C(C2(COC)CC2)=O)CCC(C2CN(C(c3cc(Cl)cc(C)c3C)=O)C2)CC1 c1(C(C(=O)NCC(CO)NC(C(C2CCC2)OC)=O)(C)C)ccccc1C c1(OC)cc(C(=O)NC(CNC(=O)CC2OCCC2(C)C)C(C)C)cc(F)n1 CCC(C)(C(=O)N(CCCCNC(=O)CC1C(=O)ON=C1C)C)C(F)F c1(OC)cnc(C(N2CCC(C(C)NC(=O)CC3CC4CC4C3)CC2)=O)c(F)c1 C(=O)(C(O)C(CCC)NC(C1CC(CF)C1)=O)NC(C#C)(C)C1CCC1 C1(CNC(c2ccoc2)=O)CCCCN1C(=O)CC1CCC(C(F)(F)F)CC1 C=CC1(C(=O)NCCC2CCC(=O)N2)CCN(C(c2ocnc2C)=O)C1 C1(C(C)NC(=O)CC2CCCC2)COCC1NC(C12CC(CO1)C2)=O CC1(C)C(C)(C)C1(F)C(N1CCC(C(F)C(=O)N2CC(Cc3ccoc3)C2)C1)=O c1(C(=O)NC2C(CNC(C=C(COC)C)=O)CC2)cc(C)cc(F)c1 C#Cc1ccc(C(=O)N(CCCNC(C2(C3CCCO3)CC2)=O)C(C)C)cc1Cl CC(C)C(C)(O)C(=O)N1CCCN(C(=O)CN2CCN(c3nncs3)CC2)CC1 Cc1ccc2c(C(=O)NC3CCN(C4CCN(C)CC4)CC3)c(C)ccc2c1 O=C(C1=CC2CCCC12)NC1CCSC12CN(C(c1ccc(C(F)(F)F)o1)=O)C2 CC#CCC(C(=O)NC1CCOC1C)NC(C1CC2(CC2)CN1C)=O c1(OCC)c(C)cccc1C.N12CCC1C(=O)N1CC(C1)CNC(=O)C2=O c1(C(=O)NCC2C(NC(C34CC(OC)C3C4)=O)CCC2)c(F)cc(C)cc1F C1(NC(c2cc(C)nn2C)=O)CC=C(C(=O)N2CCCC2CCN(C)C)C1 C1(CC(NOCCC#C)=O)CC2(CC2)CN1C(c1ccoc1Cl)=O C12(C(=O)NCCS(CC)=O)CCCC1CN(C(c1cn[nH]c1)=O)C2 C1(C(=O)NCC2C(C(=O)NCCN3CCC(OC)C3)CC2)CCC=CCCC1 Cc1cc(N)c(C(=O)NC2(C)CC(NC(c3cc(C)n(C(F)F)n3)=O)C2)cc1C CN(CCN1CCCCCC1)N1CC2(CCN2c2ccccc2)C1 C=CC(CC)CC(=O)NC(C1(C(N2CC(O)(C(=O)OC)C2)=O)CC1)C C1(F)(CNC(c2c(CC)onc2C)=O)CCCN(C(C2CC=CCC2)=O)C1 C1(NC(CC)=O)CC(CNC(=O)C=Cc2cnc(C)s2)C12CCC2 CC1(c2cn(CCN(C)C)nn2)CCCN(C(c2cnn(-c3cccnc3)c2)=O)C1 c1(NC(C2C(CNC(CC(C)=C(C)C)=O)CCCC2)=O)cncc2ccccc12 C(N=c1[nH]ccnc1F)C1(C)CC(NC(C2CC(O)(c3ccncc3)C2)=O)C1 c1(C(=O)NC(CCCC)CO)cnc2c(c1)CCN(C(c1csnc1C)=O)C2 c1(C(=O)NCCC2(NC(C3COC(=O)C3)=O)CC2)ncc2ccccn12 c1(C(=O)NC2CC(F)(CNC(C3C4CCC(F)(F)C34)=O)C2)ccn2cncc2c1 c1(C(=O)NC2CCC(C)(CNC(c3nc(=N)cc[nH]3)=O)C2)cn2ccccc2n1 C(CC1CCCc2ccccc21)(c1n(C)nnn1)NCc1ccco1 CS(=O)(=O)c1csc(C(N2CCCSCC2c2ccccc2)=O)c1 C1(CNC(=O)C=C2CCC2)CC2CCC1N2C(=O)CC1(O)CCC1 C1(NC(CSCC=C)=O)CC=C(C(=O)NC2CC(CCOC)C2)C1 C(C(CC(F)(F)F)NC(C12CC(C)(CO1)C2)=O)NC(c1c(C)nccc1)=O O=S(=O)(c1cccc(Cl)c1)N1CC2(CCC(Nc3ncnc4n[nH]c(Br)c34)C2)C1 CC(CCC(F)(F)F)NC(C1(CNC(=O)CN(C)C(N)=O)CC1)=O CC(C)CCCC(C)C(=O)NC1CN(C(=O)CCCC(C)(F)F)CC1C CCC(CC)C(=O)N1CCNC(C(=O)NCc2ccc(-c3ccncc3)cc2)C1 CC(CC(=O)NCC(C)(CO)NC(c1cc(Cl)c[nH]1)=O)CC(C)(C)C C(C(O)CCNC(=O)C(C1CCCC1)N(C)C)NC(C1(CC(C)C)CC1)=O C=CCC(C(=O)OCC)NC(=O)COCCNC(C1CC12CCCC2)=O C1(C(N(C)CC=CC(N2CC(F)(CO)C2)=O)=O)CCC2(CCC2)C1 C#CCCCCC(=O)NC1COCC1NC(c1oc(Br)cc1C)=O Cc1n[nH]c2cc(C(=O)N(C3CN(C(c4ccon4)=O)CC34CC4)C)ncc12 N1(C(CCNS(CC)(=O)=O)=O)CCC(NC(C2CCC(=O)N2C(C)C)=O)C(F)C1 C(=O)(CCC(=O)N(C)CC1CCN(C(=O)CP(C)(C)=O)C1)Nc1nnc(C)s1 C1(CC)CCN(CC)CC1.n12cc(nn1)C(=O)NCC(C1CC1)NC(=O)C21CC1 C1(CCNC(C(CC)NC(C)=O)=O)COCCN1C(c1cn(CC)cn1)=O Cc1csc(C(N2CCC(CN(C(=O)COCCN(C)C)C)C2)=O)c1C c1(C(=O)NCC2CCCN(C(c3ccc(C(F)F)nc3)=O)C2)c(O)cccc1Cl c1(N(CC(CCCC)O)C)cc(CO)cc(C(F)(F)F)n1 C12(CNC(C3N(CC)CC3)=O)CC(CN1C(=O)C(F)CC1CCCCC1)C2 O=C(C1c2ccccc2CN1Cc1cnc2ccc(Cl)cn12)N1CC(O)C(O)C1 C(C(C)(CO)CN=c1cc(C)nc(N2CCC(NC(CCO)C(F)F)CC2)[nH]1)OC C12(C(=O)NCC(CCOC)O)CCCC1CCN2C(c1cc([N+](=O)[O-])c[nH]1)=O N1(C(C2N(C(CCCC#C)=O)CC(O)C2)=O)CC2(CCC(=O)NC2)C1 c1(CN2CCC(N(C(c3cnc(N(C)C)c(Cl)c3)=O)C)C2)c[nH]c2cccnc12 N1(C(C(C)=CC)=O)CCCC(C2CCN(C(c3ccc(N)cn3)=O)C2)C1 C1(CC(=O)NCC(CC)C#N)CN(C(=O)CC2(COC)CC2)CCO1 c1(C(=O)NCC2(CN(C)C(c3cnc(N)c(Cl)c3)=O)CC2)n[nH]c2c1CCC2 n1(CC)c2ccccc2c2cc(CC3CN(c4ncc(S(C)(=O)=O)cn4)C3)ccc12 C1(N(C(C(C=C)C)=O)C)CN(C(=O)CC(c2cccc(F)c2)O)CC12CC2 N1(C(C(c2ccccc2)NC(C)=O)=O)CCC12CCCN(C(=O)C(O)C(C)C)C2 Cc1cc(Br)ncc1CNC(=O)C(N1CCC(OC(C)(C)C)C1)=O N1(CC(=O)N(CCN(C(=O)CC2CCCOC2)C)C)CCC(F)(F)C1 C=CCC(C)(C)C(=O)NCC1CC(C(=O)Nc2cc(C)cnc2O)CO1 CC(C)(CCC(=O)NC1CNC(=O)C1)NC(=O)CC1(O)CCOC1 N1(C(C)=O)CCC(N(C(CCNC(CNC(N)=O)=O)=O)CC(F)F)C1 c1(Cn2c(C3(NC(CC)C(C)C)CC(C(C)C)C3)nnn2)nn(C)cc1Cl C1(NC(CC2CN(C(c3cn(CC)nc3)=O)C(C)C2)=O)CCC(C2CC2)C1 c1(N(C(Cn2c(CCC)ncc2)=O)C)cc(NC2CN(CC)C2)ncn1 N1(C(CC2(C)CCN2C(=O)COC2CC=CC2)=O)CC(F)CC1CO C1(C2(C)CC2)(NC(C=CC(C)NC(=O)CC2CCCOC2)=O)CC1 N1(C(C(C(CC)CC)OC)=O)CCC2(CCC(NC(C3CCNC3=O)=O)C2)C1 N#CC1CCC(C(=O)NC2CC(CNC(c3ccc(C(F)(F)F)nc3)=O)C2)C1 C1(NC(c2ccc(P(C)(C)=O)o2)=O)CCN(C(=O)Cc2cnc[nH]2)CC12CCC2 C1(NC(C2CC(OC)C2)=O)CN(C(=O)Cc2nocc2C)CC12CCOCC2 N1(C(c2cc(OC)n(C)n2)=O)CCN(C(c2c(F)cc(C)cc2F)=O)CC1C#N Nc1c(C(=O)OCC(=O)Cc2ccccc2Br)cc(F)c(Br)c1F c1(NC2CCC(=O)NC2)ccc(S(=O)(=O)NCCCc2nncs2)c(Br)c1 c1(CC(=O)N(CC(C)NC(C(C)(C)OCC)=O)C)cccc([N+](=O)[O-])c1 C#Cc1cncc(C(N2CC3CCC3(CNC(c3cocn3)=O)C2)=O)c1 C(=O)(C(N)CCCCC#N)N1CCC(Br)=C(C)C1 C1(C)(CNC(C(=Cc2ccncc2)C)=O)CN(C(c2cnc(Cl)n2C)=O)CCO1 C1(NC(CS(=O)(=O)NCC)=O)CC2(C1)CN(C(=O)CCC13CCC(CC1)C3)C2 N1(C(c2ccn(CCC)n2)=O)CC2CN(C(=O)CN(C)C(N)=O)CC2(C)C1 c1(C(C)OCC(C)C)noc(COC(c2cnnn2-c2ccccc2)=O)n1 C1(N2S(=O)(=O)CCC2)CCN(N2CCC(c3ncccc3F)C2)CC1 N1(C(C2CN(C)C(=O)C2)=O)CCC(C2CC2)(CNC(c2ccc(F)cc2)=O)C1 C1(N(C(CN(C2CC2)CC)=O)C)CN(C(=O)CC2CCCC(C)(C)C2)CC1(C)C c1(C(=O)NC2CCCC2NC(=O)C(F)CC2CCCCC2)cnc(C2CC2)nc1 Cc1ccc(C(=O)NC(CO)C(C)NC(=O)CCC(F)F)cc1OCC(F)(F)F Nc1ccc(C(N2CCOCC2CCNC(=O)C(O)C(F)F)=O)c(F)c1F N1(C(Cc2c(C)n[nH]c2)=O)CCCC(CCNC(=O)C(c2cccnc2)C)CC1 C1(CCC(=O)NC(C2CC(F)(F)C2)C)CCCN1C(C1CC1(F)F)=O Cc1ncnc(C)c1CC(=O)NCC1CC1NC(C1CCCN1C(=O)C1CC1)=O c1(CC(=O)NCC(CCOC)NC(CS(CC)=O)=O)ccc(OC)c([N+](=O)[O-])c1 Cc1c(C(=O)N(C(C)CNC(=O)Cc2cnccn2)C)ccc2c1NC(=O)C2=O C(=O)(C1CCCc2cc(O)ccc21)N(CC(CNC(C(CC)F)=O)(C)C)C c1(C(=O)NCC(N(C)C(C2(C)CCSCC2)=O)C2CC2)cc(=O)cc(Cl)[nH]1 C1(NC(c2c(O)ccc(C)c2)=O)CCCCCN(C(C2CN(S(C)(=O)=O)C2)=O)C1 CCC(C)(C(=O)N1CCCN(C(c2nc(C)ncc2Cl)=O)C(C)C1)C(N)=O O=S(=O)(c1ccc(Cl)cc1)N1CCN(c2nnnn2CC2CC=CCC2)CC1 c1(NC(C2(F)CN(C(=O)CCOCC(F)F)C2)=O)cncc(OCF)c1 CCC(COC)C(=O)NCCN(C(=O)C(CO)c1ccccc1)C1CC1 c1(C(C2CCCCC2)=O)cccc(NC(N2CCC2C2CCOC2)=O)c1 N1(C(COCCC)=O)CCCC2(CNC(C3CC4(C3)CC(F)(F)C4)=O)CCCC12 c1(NC2(CNC(c3[nH]cc(C#N)c3)=O)CCCC2)ccc(Br)cc1[N+](=O)[O-] N1(C(CCCCOCC)=O)CC2CC1CN2C(=O)CNC(N)=O N1(C(C(CC2CN(C(c3cccc(C)c3)=O)C2)F)=O)CCC2(CC1)CC2C#N C1(C(=O)OC)CCCC(NC(Cc2ccc(CNC(C3(C(N)=O)CC3)=O)[nH]2)=O)C1 C(=O)(C1=CCCOCC1)N(C(C(=O)NC(C(C)C)c1ncc[nH]1)C)C1CC1 C1(CNC(C(C)OC)=O)CC2(CC(NC(c3cc(Cl)c(Cl)n3C)=O)C2)C1 N1(c2ccc(C)cn2)CCC2(CC1)CC2C(=O)NCC(Cc1ccccc1)CO O=C(N=c1cco[nH]1)C1CN(Cc2cnc(Cl)nc2)CCS1 N1(C(C(c2c(OC)cccc2)OC)=O)CC(NC(=O)COCCF)CC1(C)C C1(C)(NC(c2cnc(CCC)s2)=O)CCN(C(=O)C(F)=CC2CC2)C1 c1(C(N(CCN(C(c2c(CC)con2)=O)CC)CC)=O)cnc2n1CCCCC2 C1(CC(=O)NCC2CC2NC(c2cc(Cl)cn2C)=O)(CC)CCOCC1 CC1=CCC(C)(C(=O)NCC(C)CNC(c2cccc(C3CC3)c2)=O)CC1 CC12CCN(C1)C(=O)O2.C12(CCOCC1)C(=O)NC2.C(C)(C)(C)OC(C1CC1)=O.N C1(c2nnnn2C(C)C)(Nc2ccc(C#C)cc2)CCCC(F)(F)CC1 c1(NC(C2C(O)CCN(Cc3ccc(N(C)C)nc3)C2)=O)cc(O)c(Cl)cc1Cl c1(C(=O)OCC)cnc(NC(C)CNC(=O)C(C(C)C)NC(=O)C(C)(C)C)nc1 C1(CNC(CSCCC#N)=O)COCCN(C(C2C=CCC2)=O)C1 c1(C(=O)OC)ccc(Cl)c(S(=O)(=O)N2CCC3(C2)CN(c2ccncn2)C3)c1 CCC(C)CCC(=O)NCC1CCN(C(c2c(C(F)(F)F)cnn2C)=O)C1 N1(C(c2sc(C(=O)OC)cc2Br)C(=O)NCCCNC)CCC2(CC(OC)C2)C1 Cc1oc2ncnc(O)c2c1C(N1CC=CC(NC(C2CCOC2C)=O)C1)=O C1(C(NCP(OCC)(C)=O)=O)CC12CCN(C(c1cncc(NC)c1)=O)C2 Cc1nccc(C(=O)NCC(C2CCN(C(C3(SC)CCC3)=O)CC2)(C)C)c1N C=CC(C)(O)CC(=O)NCC1CC(c2ccccc2)C1.C1(=O)C(F)CC2CN1C2 Cc1scc(C(N2CC(NC(c3c(C)ncn3C)=O)C2)=O)c1C1CC1 C1(C(N2C(C(=O)NC(c3cnc(C)s3)C)CC(O)C2)=O)CC(=O)NC(C)C1 C1(CCNC(CC2(N(C)C)CC2)=O)CCCN(C(c2ccc(=N)[nH]c2)=O)C1 N1(C(c2c(COCC=C)ccs2)=O)CCC(CO)(NC(=O)C(c2cnn(C)c2)=O)C1 c1(C(=O)NC(C(CO)NC(C2ON=C(C)C2)=O)C)cn(C)nc1-c1cnccn1 c1(OC)ncc(F)c(=NC2CCN(C(c3ccc(OC(F)F)cc3)=O)CC2F)[nH]1 c1(C(N(C2CCCC(NC(Cc3nccc(C)c3)=O)C2)C)=O)cccn(C)c1=O C1(N(C(CC(C)OC)=O)C)CCCC2CN(C(c3cc(C)nc(O)n3)=O)CC12 CCCC(CC)C(=O)NCC=C1CCN(C(=O)COCc2nc(C)no2)CC1 N1(C(c2c(SC)ccs2)=O)CC2CC2(CNC(C2CCC(=O)N2C)=O)C1 C1(C)(C(=O)NCC(C)CCO)C=CCN1C(c1cn(C)cn1)=O N1(C(C(=O)NC2CCCC(C(C)(C)C)CC2)=O)Cc2cc(O)nnc2C1 C1(CCNC(c2cc(Cl)cnn2)=O)CCCCN1C(=O)CC1C=CS(=O)(=O)C1 c1(C(=O)NCCC(CNC(c2c(OC)cccc2)=O)(C)C)cccn(C)c1=O C1(NC(=O)NC2(c3cccc(Cl)n3)CC2)CN(CC(F)F)CC12CCOC2 Cc1ccc(C=CCCNC(=O)NCCCCC(C)C)cc1 c1(C(C)(C)C(=O)NC2(NC(=O)CC3CC(F)C3)CC2)cc(Cl)cc(Cl)c1 c1(Oc2cc(Cl)nc(C3CC3)c2)cnc2nccn2c1 C(CCCCC(=O)NC(C)(C)CNC(c1ncc(C(F)F)s1)=O)OC C(=O)(CCC(CC)NC(=O)COCC(C)(C)C)NCC1(C=C)CCC1 c1(N2CCN(CCC)CC2)nc(=NCC(O)(CC)CC)[nH]c2c(F)cc(F)cc12 c1(CNC(C(C)NC(CC)=O)=O)ncccc1OCCF.C12CC1C(=O)N2 c1(C(=O)NC(CC)CNC(=O)CCOCC2CCCO2)ccc(COC)nc1 C1(NC(=O)C=Cc2cc[nH]n2)CC(O)CN(C(=O)CCOCC(F)F)C1 c1(OC)ccc(-c2ccc(C(=O)NCc3ccc(O)c(Br)c3)nc2)c2cn[nH]c12 N1(C(C(C)S(C)(=O)=O)=O)CC2CCCC(NC(c3cc(CO)on3)=O)C2C1 C1(N(C)C)(C(N2CCC(c3cn(Cc4ccccc4)nn3)CC2)=O)CCCOC1 C1(CNC(C2C(C(=O)OC)C2)=O)CCCCC1NC(c1ccn(C)c1)=O CC1=C(C(=O)NC2CC(NC(c3cnoc3C)=O)C2)CCC(C)(C)C1 c1(C(N2CCC(C(C)NC(C(c3ccc(C)s3)C)=O)C2)=O)ccc(Cl)cc1N C(c1cnc(C)s1)=CC(=O)NCC(CC=C)NC(=O)C(Cc1ccccc1)OC C1(F)(CNC(C2CC2Br)=O)CCN(C(c2cncc(-n3cnnn3)c2)=O)CC1 c1(C(=O)NCCCN(C(C2ON=C(C)C2)=O)CC2CCCC2)ccc(F)c(Cl)n1 C(=O)(C(C(=O)NC(C)(C)C(C)NC(=O)CCc1ccc(Cl)cc1)OC)OCC N1(C(C(CC#C)C)=O)CCN(C(C2CC2CF)=O)C(CCOC)C1 C1(CCN(C)C(C2CC2c2cccnc2)=O)CCN(C(=O)C(F)(F)C2CC2)CC1 C1(NC(C(CC)(C)O)=O)CCCN(S(=O)(=O)c2cn[nH]c2)CC1 c1(C(C)C(=O)NC2CC(CCNC(=O)CC3CC3)C2)ccc2c(c1)OCO2 c1(CCC(=O)NC(CCNC(c2c(OC)cccc2)=O)C)nc2ncccn2n1 c1(C(=O)OC)cc(C)c(C(=O)NC2CN(C(c3csc(C(F)F)c3)=O)CC2C)o1 c1(C(C)NC(=O)C=CC(C)NC(=O)CSC(F)(F)F)cnn(C)c1 CC12COC(=O)N1CCN(Cc1ccc(-c3ccc(C=O)cn3)nc1)C2 C(CCCC(=O)NC1(C)CCCC1C)NC(c1n(C(C)C)ccn1)=O C1(CC=C)(NC(=O)COC2CCOCC2)CCN(C(C2(CN(C)C)CC2)=O)C1 c1(SC(C)C)ncccc1C(=O)N(C)CC1C2CN(C(C3CCCCO3)=O)CC12 c1(C2C(C(=O)NCC(N(C(=O)CC3(C)CCC3)C)C3CC3)C2)cccnc1 CC(CN=c1[nH]c(=NCCN2CCCOCC2)[nH]c2ccsc12)c1ccncc1 N(C(=NCC1COCc2ccccc21)NCC)CC(CN1CCCC(CC)C1)C C1(NC(c2c(C)csc2)=O)CCC(C)N(C(=O)COCCC(C)C)C1 c1(C(N2CCC(NC(c3ccc(C)c(O)c3)=O)(CO)C2)=O)ccc(S(C)(=O)=O)s1 c1(C(=O)NC(CC)CNC(=O)C(C2CCCCC2)N(C)C)ccc(=N)[nH]n1 C1(C(N2CC(c3ncc(C)o3)C2)=O)(COC)CCN(C(=O)Cc2nocc2C)C1 C1(C)(C(=O)NCC(C)NC(c2ccc(-c3ccccn3)o2)=O)CCN(C(N)=O)C1 C1(CC(=O)NCC2(NC(=O)CN3CCSCC3)CC(F)(F)C2)CCCCC12CC2 C12(CNC(C(C)OCC#C)=O)CN(C(c3cnccc3OC)=O)CC1CCO2 N1(CC(=O)NCCn2cncn2)CCC(O)C(C(=O)NCC=C2CCOCC2)C1 C(C(C)C(=O)N1CC(CC(C)NC(=O)CCCc2ccsc2)C1)SC c1(C(=O)NCC2C(C)C2)ccc2c(c1)NC(=O)CCC2 c1(OC)ccc(F)c(CC(=O)NCCC(C)NC(C2C3CCN2CC3)=O)c1 c12cc[nH]c1C(=O)NCCC1CCN(C1)C2=O.c1(CN(C)C)cn[nH]c1 Cc1ccc(SCC(=O)NC(CNC(c2cc(O)ccc2C)=O)CO)cc1C C(=O)(CC1CN(C)c2ccccc21)N(C(CCNC(CCSC)=O)C)C c1(C(N2CCC3(CCC3)C2)C(=O)NCCCCCC)cc(C)c(F)cc1Br n1(CC=C)nnnc1C(C1CCCOC1)NCC1(C2CCCCC2)CCCC1 CCC(CC(=O)NC(CNC(c1csc(Cl)n1)=O)(CC)CC)OC C(=O)(C(C)(O)Cc1ccccc1)NC(C)CCNC(C1(c2cnn(C)c2)CC1)=O c1(COC)nnc(CNC(=O)C(=O)NC(C2CC(C)(C)C2)CO)s1 c1(C(=O)NCC)ccc(-c2ncn(C)c2CNCCC2CCCOC2)cc1 c1(C(=O)NCc2cc(C(N3CC(C(N)=O)C(C(N)=O)C3)=O)sc2)cnc(O)nc1O C1(N(C(=O)COc2ccccc2)C)CCN(C(c2ccncc2O)=O)CC12CC2 CC(CC(=O)NC1CN(C(=O)CC(C(F)F)c2ccccc2)C1)C(F)(F)C(F)(F)F c1(OC)cc(Cl)ccc1COC.c1(C2C3(CCC3)N2)nnnn1C1CC1 CON(Cc1ccccc1)C(=O)COC1CN(C(=O)CN(C)C2CC2)C1 n1(CC(=O)NC2CCCN(C(Cc3nc(C)c(C)s3)=O)C2)cc2ccccc2n1 C1(C(C(=O)N(C(c2ccccc2)CNC(C2(N=[N+]=[N-])CC2)=O)C)O)CCCCCC1 C(=O)(C(CCCCCC)N(C)C)N(CCCNC(C1(CC=C)CCOC1)=O)CC c1(OC)cccc2c(NCC(c3ccccc3OC)(C)C)c([N+](=O)[O-])cnc12 N1(C(Cc2scc(CC)n2)=O)CCC(C(N)=O)(NC(C2CSCC(=O)N2)=O)CC1 C1(NC(CSCCCC)=O)CCCC1C(C)(C)C(=O)NCC1(CC)CC1 C1(C)(COC)CC(NC(=O)C=C2CC2)CN1C(=O)CCc1ccc(F)cc1 C(C(C)(C)C(=O)NC1COCC1C(=O)NCC(C)C#N)SC c1(OC)c(C(=O)NCC2CC(NC(=O)CNC(N)=O)CCO2)csc1Cl N1(C(C(CSC)C)=O)CC2CC2(NC(c2cnn(-c3cccc(Cl)c3)c2)=O)C1 N1(C(C=Cc2ncc(C)[nH]2)=O)CCCC(C2CN(C(=O)C(C)(C)C(C)(F)F)C2)C1 N1(CCCc2ccc(C)cc2)CC(NC(c2conc2C)=O)C(C)(C)C1 N1(C(C2N=C(C)SC2)=O)CC2CCC1C(CNC(c1cnc3ccsc3c1)=O)C2 C(=O)(CCC(=O)N1CCC(CC(C)NC(=O)C(N2CCCC2)C2CC2)CC1)OC C1(CNC(CCOC)=O)CN(C(C2CC2F)=O)CC1OC1CCCCCC1 CCC(CC)C(C)C(=O)N1CC2(C(N3CCCC(C(=O)NC)C3)=O)CC1CO2 Cc1cc(C(=O)NCC(C)(C)CNC(=O)CSc2cnn(C)c2)cc(O)n1 c1(C(=O)NC(C2CCN(CC(N)=O)CC2)C)cn2ncsc2n1 C(N=c1[nH]c(N(C)CCOCCO)nc2c1COC2)C1(CCC)CCC1 c1(CC(N2CCN(C(CNC(N)=O)=O)CC2C2CC2)=O)cc[nH]c2nccc1-2 N1(C(CNC(=O)NC)=O)CCC2(CC1)CC2C(=O)NCC(C)(O)C(F)(F)F n1(CC)cnc2nc(=NCC(C)(C)C(C)C)[nH]c(NCCCCCOC(C)C)c12 C(=O)(C1=CCC(NC(C2(CC3CC3)CC2)=O)C1)NC(CC#C)CC c1(C(=O)NC(CN(C(c2cc(CO)ccn2)=O)CC)C)ccc(S(=O)(=O)NC)o1 c1(OC)ccc(C(=O)NCC2CN(C(=O)C(=O)NC3CC3)CCC2C)nc1Cl CC(C(=O)N1CCCC(N(CCO)C(c2cc(=O)n(C)o2)=O)C1)P(C)(C)=O c1(CC(=O)NCC(CC=C)NC(c2ccoc2Cl)=O)ccccc1CC(N)=O c1(C(=O)NC(CNC(C(CCC)N(C)C)=O)C(C)C)cc(Br)cc(C)c1N C#CCCC(O)CCNC(C1(C)C=CCN1C(C1CCOCC1)=O)=O N1(C(CC=CC=C)=O)CCC(CF)(NC(=O)C(C)(C)c2ccccc2)C1 O=C1CCC(C(=O)NCCCN(CCO)C(C2CCCS2)=O)C1 c1(C(=O)NCC(CNC(=O)CC2CC2)O)oc(C2CC2)nc1C(F)F C1(N(C(=O)CCC2CCCC2)C)CCN(Cc2cncs2)CC1 c1(C(=O)NCC(C2CCC2)NC(C=C(COC)C)=O)oc(S(N)(=O)=O)cc1C c1(CC(=O)NC2C=CCN(C(C(=COCC)C#N)=O)C2)cccc2ccccc12 C1(NC(CCC(=C)Br)=O)CN(C(=O)Cc2cnc(C)[nH]2)CCC1O c1(C(=O)NC)ccc(NCC(C2CC2)NC(=O)CN(C)C)c([N+](=O)[O-])c1 C(=O)(N=c1[nH]oc2cccnc12)C1C2CN(Cc3cnc(OC)c(Br)c3)C1C2 CC1CCN(C(C2CC(OC(F)F)C2)=O)CC1NC(=O)C#CC(C)(C)C c1(OCCC)ccc(C(=O)NCCCN(CCO)C(C2CCC(F)C2)=O)c(C)c1 c1(C(=O)NCC2C(NC(c3c(C)ncn3O)=O)CCCC2)cc(Cl)c(Cl)n1C c1(C(N2CC3CC2CS3)C(=O)Nc2c(C)cccc2)cc(F)c(Cl)cc1F C1(CNC(CCOCCC)=O)CC2(CN1C(=O)CC(=O)OC)CC2(F)F c1(SCCC(N2C(CNC(CCOCC)=O)CC2)=O)ccc(F)c(F)c1 N1(C(c2c(CC)noc2)=O)C2CCC1CN(C(=O)CC1CC(OC)C1)CC2 C#Cc1ccc(C(N2CC3CCCC2CN3C(C2CCC=CCC2)=O)=O)cc1F C1(N(C(C23CC(c4ccccc4)C2C3)=O)CC)CCN(C(=O)CN2CC3CC3C2)C1 Cc1ccc(CC(=O)N(CCNC(C2CCN(C)S2(=O)=O)=O)CC2CC2)cc1Cl Cc1ccc(-n2cc(NC(=O)CN(C(=O)CCC3CC(F)(F)C3)C)nn2)cc1 C(=O)(C(C)(F)C(=O)NC(CO)C(C)NC(=O)CC1(C2CC2)CC1)OCC N1(C(CCOCC#C)=O)CC(C2CN(C(=O)C(F)C(F)(F)F)C2)C1 C1(N(c2c(C(=O)OCC)csc2)C(C2CCCC2C)=O)CC2CC1CN2 c1(CC(=O)N(CC(C)NC(C)=O)C(C2CCN(C(CC)=O)C2)=O)ccc(F)c(Cl)c1 CC(C)(C(=O)NCC1(F)CCCN(C(C2CC(=O)N(C3CC3)C2)=O)C1)C(F)F c1(CC(=O)N(C2CCCN(C(C3(C)CCC3)=O)C2)C)cnn2c1CCCC2 C=CCC(C)(C)CC(=O)N1CC(O)(CNC(=O)CSC2CCOC2=O)C1 CCCC(C)CC(=O)Nc1cccc(NC(=O)COc2cccc(C#N)c2)c1 CN1CC(C(N2CCC(CNC(=O)CCn3cnnn3)C23CC3)=O)CCC1=O c1(NC)c(C(=O)NC(C)CNC(=O)COC(C)C)cccc1F C1(CC(=O)NCC(=O)NCC#C)CCCCC1N c1(SCC)cnc(O)c(C(N2CCC(CCNC(=O)C(C)(O)C3CCC3)C2)=O)c1 C(=O)(C(CC)c1cccnc1)N(C1CCCC1)CCCNC(C=CCC)=O N1(C(c2cc(C)[nH]c2C)=O)CC(NC(c2cccc3nn[nH]c23)=O)C2(CCC2)C1 c1(CC)nc2ccc(Cl)cn2c1C(=O)NCC12CC1CN(C(=O)C(C)S)C2 N1(C(C2(CC)CC2)=O)CC2CC(O)C1C2NC(=O)COc1cccc(N)c1 N1(C(c2ccc(C)o2)=O)CCN(C(=O)CC2CCC(C)(C)O2)CC1C Cc1cc(C)c(NC(C2CCCC2NC(=O)CCCN(C)C)=O)c([N+](=O)[O-])c1 C1(c2ccccc2)(C(=O)NC(CNC(c2csc(O)n2)=O)CO)CCOCC1 C(CN=C(NC1CCC1)N1CCC(c2nncs2)C1)(c1cccs1)N(C)C c1(NC(C2(F)CN(C(C3CC(N4CCCC4)C3)=O)C2)=O)ccc(C(=O)O)s1 c1(C(=O)NCC(C)CNC(=O)C(C)CN(C)C)cnc2c(c1)N(C)CCO2 Cc1nc(C)c(C(N2CC3CC3(CNC(=O)CCOCC(F)(F)F)C2)=O)s1 C1(C(=O)NCC2CCCC(CNC(c3ccon3)=O)C2)CCCNS1(=O)=O C(C)(CNC(c1csc(C(C)OC)n1)=O)(CC(C)C)NC(C(CCC)=CCC)=O C(=O)(C1=C2CCCN=C2NN1)NC1CC(NC(C(CC=C)CC=C)=O)C12CCC2 C#Cc1ccc(CCC(=O)NCCC(C)(C)NC(C2CCN2C)=O)cc1 Cc1cc(=NCCN(C)C)[nH]cn1.c1(CCNCC2CC2)cccc2ccccc12 Cc1c(CCC(=O)NC2CC(NC(c3nc(=N)cc[nH]3)=O)C(O)C2)cnn1C Cc1nc2nccc(N3CCC(F)(CNC(c4cc(C)c(C)nn4)=O)CC3)n2n1 c1(CSc2nccc(C(=O)OC)c2)ccc(Br)nc1Cl c1(C(c2nnnn2C)NC(C=C)C2CCC2)cnn(C)c1Cl C1(NC(c2cccn2C2CC2)=O)CC2CCC1C(NC(c1coc(O)n1)=O)C2 c1(NC(CC)=O)cccc(C(N2CCOC(CNC(C3OCC3(C)C)=O)C2)=O)c1 C(=O)(C1CCc2c(Cl)cccc21)NCC(C)N(C(c1nccn1C)=O)CC Cc1cc(O)ncc1C(=O)NC1CCCCC1CNC(=O)Cc1cc[nH]c(=N)c1 N1(C(CCCSC)=O)CCC(CN(C(=O)CCOCC2CCCO2)C)CC1.O c1(C(N2CCOCC(NC(C(C3CCC3)OC)=O)C2)=O)c[nH]c2cc(C)ccc12 c1(C(N2CCN(C(C(=Cc3cccnc3)C)=O)C(C)C2)=O)cccc2sccc12 N1(C(C(CC)n2cncn2)=O)CC(NC(c2cccnc2C)=O)CC1C N1(C2C(=O)NC3CC23)CCC12CCC(C)(C)CC2.c1(CC)cc(OC)ccc1Cl CC(C)C(C)(CNC(=O)CSCCN(C)C)NC(C1CC=CCC1)=O N1(C(c2c(C)onc2O)=O)CC2CCC(C1)N2C(=O)Cc1ccccc1[N+](=O)[O-] c1(C(N2CCCC(COC)CC2)C(=O)NCCCCCC)cc(OCC)ccc1Br c1(OC)nccnc1C(N1CCC(C(C)C(=O)NCc2nc(C)cs2)C1)=O C1(CC(=O)NC2(c3nc(C)[nH]n3)CC2)C2CCCC2N1C(C1CC12CCOC2)=O c1(C(=O)NCC(CNC(C(C)CN(C)C)=O)C(F)(F)F)c(Cl)ccc(Cl)c1O CC1CN(C(c2nccn2C)=O)CC(C)N(C(c2ccc(C3CC3)s2)=O)C1 CC1CN(C(=NCCC2CC3C=CC2C3)NC2CC2)CCC1O C(=O)(C(C)(C)CS(N)(=O)=O)N1CCC(C)(NC(COCc2c(C)cccc2)=O)CC1 C1(C(N2CC(N(C(=O)CCC3CC3)C)C2)=O)CC1C1CCCC1 N1(C(CSCC#C)=O)CC(NC(C2CCCS2)=O)C2(CCS(=O)(=O)CC2)C1 c1(CC(=O)NC(CC)(C)CNC(=O)Cc2c[nH]nc2O)cnc2n1CCCC2C Cn1nc(O)cc1C(N1CC(CCCCNC(=O)Cn2ccnn2)C1)=O n1(CC(=O)N(CC(C)OC)C(C)C)cc(C(=O)OC)nn1 N1(C(C(C(=O)NC)(C)C)=O)CCC(C2CCN(C(=O)CCC3CC3(C)C)C2)CC1 c1(NCc2nc(C(=O)OC)sc2)ccc(OC(F)(F)F)c(NC(C)=O)c1 N1(C(COCC#C)=O)CCC(CN(C)C(C2CN(C(c3cccs3)=O)C2)=O)C1 c1(C(=O)NCCCCCN(C(=O)CC2CCCCC2)C)c(F)cncc1Br N1(C(C(C(CC)O)C)=O)CCC2(CC1)C(NC(=O)CCC(C)N(C)C)CS2(=O)=O c1(SC)cscc1C(=O)NCC1(NC(c2cscn2)=O)CCOC1 CC(C)C(O)C(=O)NCC=CCNC(=O)CSc1nncs1 N1(C(C2CN(C)C2)=O)CC2(CCC2NC(c2occc2Cl)=O)C1 Cc1ccc(NC(=O)CN(C)C(C2CCC(=O)N2)=O)cc1C N1(C(c2nc(C)sc2)=O)CC(CNC(=O)CN2CC3CCC2C3)CC1(C)C C(=O)(CCCC(=O)NC(CNC(C1(C)CC2CC2C1)=O)CCOC)N(CC)CC c12nc(C)c(s1)C2.C(c1ccc(C)s1)=CC=O.N12CC=CC1C2.C1=CC=C1.CC=C Cc1ccc(CCC(=O)NCCCNC(C2CCC(O)CC2)=O)cc1C C1(C(=O)NC2C(C(N3CC(CCC#C)C3)=O)OCC2)CCC(N=[N+]=[N-])C1 Cc1c(N2CCC2C(N2CCOCC2)=O)ccc(-c2ccc(C3CC3)cc2)c1F CC(N=c1nc(N(CC(C)(C)CO)C)c2c([nH]1)CCOC2)c1ccccc1Br C1(C(C(=O)NCC2CCC2)N(CC(Cl)Cl)C)CCC(c2ccccc2)CC1 Cc1c[nH]cc(C(N2CCC(C(C(C)C)NC(C3CCC(C)O3)=O)CC2)=O)c1=O CCCC(C)(C)CC(=O)N1CC(CN(C)C(C2(O)CC(CF)C2)=O)C2(CC2)C1 C1(CNC(C(CCCC)F)=O)CN(C(=O)CCC(C)C)CC(C)(C)O1 C1(CNC(=O)CNC(=O)C(F)(F)F)CCCC2(CN(C(=O)C(F)C3CCC3)C2)O1 c1(NC(CNC(C)(C)C(N2CCCCCC2)=O)=O)ccc2cc[nH]c2c1 C1(C(=O)NC(C2(O)CN(C(C(C)O)=O)C2)C)CN2CCN1CC2C c1(C(=O)NCc2ccc(CNC(C3CC(C)OC3)=O)cc2)cccc2oncc12 C1(NC(C(C)=C(C)C)=O)CC2CN(C(=O)C=Cc3ccc(F)cc3F)CC2C1 c1(COC)ccnc(C(N2CCCC(CCNC(C3CC4(C3)CC4F)=O)C2)=O)c1 C(C(C(C)(C)C)NC(=O)CC1CC(O)C1(C)C)NC(C1(CC#C)CC1)=O N1(C(c2cc(OC)cc(F)c2)=O)CCc2nn(C)c(C(=O)N(C)CC#N)c2C1 c1(C(c2n(CC)ccn2)O)ccc(NOCc2ccc(Cl)cc2)cc1 C(=O)(C(CC)CCCCC)N1C(C(=O)Nc2cn(CCC#C)nc2)CC(F)(F)C1 c1(OC)ccc(CN2CCCC2CC(=O)Nc2ncccc2OC)cn1 C(=O)(C(CC(C)C)C(N)=O)N1CCCC(CCNC(Cc2c(C)con2)=O)CC1 C1(C(=O)NC)Cc2ccccc2CN1C(=O)CC(C)n1ccc(C)n1 C(C1CCN(C(c2occc2CC)=O)CC1)=CC(=O)NC(CC=C)CO Cc1c(C(=O)NCCOCCNC(=O)C(O)C2CCC2)ccc(Cl)c1Cl Cc1ccc(C(N2CCCC2CNC(C23CC(C#N)(C2)C3)=O)=O)c(F)c1F N1(C(c2c(Cl)c(C)n(C)n2)=O)CCC(CNC(C2CCC(F)(F)C2)=O)C12CCC2 C12(NC3C(O)CCN(C)C3)CCCN(C(=O)OC(C)(C)C)C1COC2 C1(NC(COC)=O)C2CC1CN(C(c1cc(N(C3CCCC3)C)ccn1)=O)C2 C(=O)(CC(F)(F)C(F)(F)F)NCC1(CNC(c2ccc(OC)cc2Cl)=O)CCC1 c1(C(=O)NCC(CC(C)C)NC(C2CCC(OC)CC2)=O)ccc(=O)n(C)n1 c1(C(C(=O)NC2CC(N(C)C(C3CC3(C)C)=O)C2)(F)F)ccc(F)cc1 N1(C(C)C)CC(NC(=O)N(C)C)CC1=O.c12cccc(c1)OC2=O C(=O)(C1CCc2nnc(C)n21)NC1CCN(C(Cc2nnc(C)n2C)=O)CC1O C1CN(C(=O)C(O)C2CNC2)CC(C(F)(F)F)O1.C(C(=O)O)=C(C)C c1(C(N(C2CCCC2)CC#C)=O)c(CNC(=O)C=Cc2ccc[nH]2)cnn1C CC1(C)CC(CNC(C2(C)CS(=O)(=O)C2)=O)N(C(=O)CC2CC3CC3C2)C1 [N-]=[N+]=NC1CCC(C(=O)NC23CC(CNC(c4ccc[n+]([O-])c4)=O)(C2)C3)C1 C1(O)(C(N2C3CC(NC(c4scc(OC)c4)=O)C(C3)C2)=O)CN2CCC1CC2 C12(C(=O)NC(C)(C)CCF)CCN(C(C3CCC4(CCC4)C3)=O)CCC1C2 c1(C(N2C(CC)CN(C(C3CCCCC3)=O)CC2)=O)nc2sccn2c1C C#CCCCC(C)C(=O)NC(Cn1ccnn1)C(=O)NC[Si](C)(C)C CC1CN(C(C2(C(=O)N(C)C)CC2)=O)C1.C1(C)(C)CNC(=O)CO1 C(=O)(C#CC1(C)CC1)N(CCN(C(=O)CC1(CO)CCOCC1)C(C)C)C N1(C(C2CCN(CCC=C)CC2)=O)CC2CCC(C1)C(=O)N2 N1(CCCCCC)C(=S)NC(c2ccnn2CC)C(C(=O)OCC)=C1C(C)F CC(C)C(C(C)C)C(C(=O)NCSc1ccccc1)N1C2CCC1CC(=O)NC2 CN1CCC(CC(=O)NCC2(CN(C)C(C3(CO)CCCC3)=O)CC2)C1=O C12(C(=O)NCC(CC=C)NC(=O)C(c3ccccc3)O)CC(C1)C(C)(C)O2 C(=O)(CCC(=O)NC)NCC(CC=C)NC(c1cccn1CC)=O C1(CC=C)(N(C(=O)CCc2cc[nH]n2)CC)CCN(C(=O)CCCN2CCCC2)C1 C(=O)(C(C(=O)NCCCNC(=O)COCC(c1ccccc1)C)C(C)C)OCC CC1CN(C(C2(CNCCNC(c3ccc[nH]3)=O)CC2)=O)CC1CC(=O)OC1CC1 CC(C)S(=O)(=O)CC(=O)NC12CC1CN(C(c1cocc1Br)=O)C2 CC1(C)CCCC(O)(C(=O)NC2CCC(NC(C3CCN3C3CCCC3)=O)CC2)C1 c1(CC(=O)O)ccc(O)c(NC(C2(C(F)(F)F)CCOC2)=O)c1 c1(OC)ccc(C(F)(F)C(=O)NC2CC(NC(c3sccc3Cl)=O)C2)cn1 C(CC(C)CCNC(C1(F)CC1)=O)NC(c1ccn(CCC)n1)=O C(N=c1[nH]c(N2CCC(CC(F)F)C2)nc2c1CCCCCC2)c1nc(Br)sc1 Cc1cccnc1C(=O)NC1(C2CCCCN2C(=O)C(N2CCSCC2)C)CC1 Cc1nc(N2CC(NC(c3cnc(C(C)C)s3)=O)CCC2C)cc(C#N)n1 C#Cc1ccc(C(=O)NC2(C(=O)NCc3ccsc3C)CC2(C)C)cc1C c1(C(=O)NCC(C)(O)CNC(=O)C=CC(F)(F)F)cc(F)cc(N)c1F c1(SCC)cccc(C(=O)NCCCC(C)NC(=O)C(C)N(C)C)c1 c12ccc(cc1)S(=O)(=O)NC2=O.C1(CCC(=O)NCCC(=O)OC)CCCN1C N1(C(CC2(NC(C3CC(=O)NC(=O)C3)=O)CCC2)=O)CCC2(CC=CCO2)C1 c12nc(co1)C(=O)N2.C(CC(C)N(C(=O)C(C)N(CC)CCC)C)NS(=O)(=O)CC C1(CNC(C2CCC2COC)=O)CC(C)N(C(=O)COCCCC(C)C)C1 CC(C)(C)CC(F)C(=O)N1CCCC1CC(=O)NC1CCCSCC1 C(=O)(C1=C(C)N(C)c2nnnn2C1C)NCC1N(C(CC=CC)=O)CCCCC1 C1(CC(=O)N(CCN(C(C)C)C(C2CCC2(F)F)=O)C)(N(C)C)CCCC1 c1(C(CC(=O)O)C2CN(C(C(CC)c3ccccc3)=O)C2)cccc(I)c1 Cc1ccn(C)c1C(N1CC(C(O)C(=O)NCC2COC(=O)N2)C1)=O C=CCC(CC(C)C)C(=O)NCCC1CCCCN1C(=O)C#CC(C)(C)O C1(c2c(CN(CC(CC)OC)C)ccs2)CC2(CSC2)C1 N1(C(c2c(CC)c[nH]c2)=O)CCC2(CCOCC2)C(NC(=O)CCNC(C)=O)C1 N1(CC(=O)N(C2CCC(NC(c3csc(F)c3)=O)C2)C)CCC(F)(F)C1 C(=O)(C(CCC1CC1)NC(=O)Cc1ccc(F)cc1)N(CC(C)O)C N1(C(C(C)C)C(=O)N(C)Cc2ccc(CO)cc2)CCSC(c2ccccc2)CC1 N1(C(C(CSC)C)=O)CCCC(NC(C2CCCC(=O)O2)=O)C1 C(=O)(C1=NNC(C(F)(F)F)C1)N1CC(O)(C(C)NC(C2CC2(F)F)=O)C1 C1(NCc2c(OC)ccs2)CCC(C)(C)CC1C C1(NC(CC(=O)OC)=O)CC(NC(=O)C(C2CCOCC2)O)C12CCOCC2 n1(C(C)C)[nH]c(C(=O)NC2CN(C(=O)C(c3ccc(F)cc3)O)CC2C)cc1=O c1(C(N2CC(N(C)C)CC(C(=O)OC)C2)=O)ccc(C#N)cc1C C1(C(N(CCC(=O)NC)C)=O)CC2C=CC1N(C(=O)Cc1n[nH]c(C)n1)C2 Cc1csc(=O)n1CC(=O)NC(C)CNC(=O)CN1CSCC1=O c1(CNC(C=C(COC)C)=O)nc(C(=O)NCC2CCC3CC23)co1 N1(CC)CCCC(C(N2CCC3CC23C(=O)NCC(=O)N(C)O)=O)C1 N1(C(C(c2ccnn2C)C)=O)CCN(C(c2cc(=O)n(C)cn2)=O)CC(O)C1 C1(CC(=O)NC2(C(N3CCC3C3CCC3)=O)C(C)C2)CCOCC1 N1(C(CC(=O)NCC)=O)CCC(NC(c2ccccc2OC2CC2)=O)C1C c1(C(=O)NC(CNC(C2C(=C)C2)=O)CC)ccc(C#N)c([N+](=O)[O-])c1 c1(C(N2CC(CC(C)NC(C3CCCC(CF)C3)=O)C2)=O)ncccc1O CON(C)C1CCN(C(c2nc(SC)ns2)C(=O)NCSc2ccccc2)CC1 N1(CC2NCCN(S(=O)(=O)Cc3ccccc3)C2)CCn2nccc2C1 C1(C2(NC(C=C(CC)C)=O)CC2)CCCN1C(=O)C(C)=C1CC1 c1(C(=O)NCC2N(C(c3n(CC)ccc3)=O)CC3CC32)ccc(=N)[nH]c1Cl C1(C(=O)NCCC(C)NC(C2CCCOC2)=O)CC2(CSC2)C1 c1(C(=O)NCCN(C(c2ccncc2C)=O)CC)cnn2c(C)cccc12 C1(CNC(C(C)c2ccsc2)=O)CC2CCCC2N1C(=O)CC1(O)CCC1 C(c1ccccc1Cl)=CC(=O)NCC(CC(C)C)NC(C1(N(C)C)CC1)=O Cc1cc(C(=O)NC(C)(CNC(c2scnc2C(F)F)=O)C2CCC2)sc1C C(=O)(CC1C(=O)Nc2ccc(F)cc21)NC1(COC)CN(C(C(CC)F)=O)C1 C=C(C)CCC(=O)NCC1CN(C(c2coc(C)c2)=O)CC1C N1(C(C(c2cccc(Cl)c2)C)=O)CCC12CN(C(C1SCCS1)=O)C2 c1(C(C)OCCNC(C2C(NC(=O)NCCO)C2)=O)ccccc1COCC C(=O)(C(C)(C)CN(C)C)NC(CNC(CCc1onc(C(C)C)n1)=O)C(C)C O=[N+]([O-])c1cccc2[nH]cc(CNCc3coc(-c4ccccn4)n3)c12 c1(C(=O)NCC(N(C(C(C)C)=O)C)C2CC2)cnc2n1CCCC2C N1(S(=O)(=O)c2ccnc3ccccc23)CCOC2(CCN(Cc3cccs3)CC2)C1 c1(CC(=O)NCC2OCCN(C(CC(COC)(C)C)=O)C2)coc2ccccc12 C1(O)(C(C)NC(c2cc(C#N)cs2)=O)CCN(C(c2sccc2F)=O)CC1 c1(CCN(C)Cc2cc(C)nc(C3CCC3)n2)ccc(C)c(C)c1C C#CCC(CC#C)C(=O)NCC1CC1CNC(=O)CN(S(C)(=O)=O)C N1(C(C(N2CCOCC2)C)=O)CCC2CN(C(c3cc(Cl)ns3)=O)CCC12 C1(NC(C(CC=CC)C)=O)CN(C(c2ccc(=N)[nH]n2)=O)C(C)(C)C1 c1(C(=O)NC2CC(N(C(=O)CC3(C)CCCO3)C)C2)cccc(O)c1F c1(C(=O)NC2CN(C(c3ccc(C(C)=O)o3)=O)C(C)CC2)cc(C)c(C)cc1N N1(C(C2(F)CC=CC2)=O)CCC(CNC(=O)C(F)(F)C(F)F)C(C2CC2)C1 CCC(C#N)(CC)C(=O)N1CC2CC1CC2NC(C1CC2(C1)CC(C)(C)C2)=O O=C1NC(CC(=O)Nc2ncc(C3CC3)s2)CO1 C1(C(=O)NCCC2CN(C(C3(Cl)CC3(F)F)=O)CCO2)(OCC)CCSCC1 O=C(CCN(CCO)C(C1SCCS1)=O)NCc1cscn1 C#CC1(O)CCCN(C(=O)C(C)N(CCC)C(C2CC(=O)N(C)C2)=O)C1 N#Cc1ccc(C(=O)NCCC(O)CNC(C2(CO)CCCO2)=O)o1 CS(=O)(=O)C(C(=O)NC12CC(C1)N(C(=O)CCC#N)C2)c1ccccc1 C(=O)(C1CCN(C)c2ccccc21)NC(c1ccc(C)cc1)CNC(=O)CO c1(C(N)=O)nccnc1C(N1CC(F)(C(=O)NCCc2cnccn2)C1)=O Cc1nc(C)n(O)c1C(=O)NC1CN(C(=O)C=Cc2cccn2C)CCC1C Cc1nc(C(=O)NCC(C(C)C)NC(=O)C=CC(C)(C)C)n(C)n1 c1(-c2c(C(=O)NC3CN(C(C(CC)O)=O)CC3F)c[nH]n2)c(F)cccc1F c1(C(=O)NC2CC3CN(C(CN(C(C)=O)C)=O)C2C3)nnn2c1CCCCC2 c1(N(C(C)CCNC(c2ccc(O)nc2)=O)C)ccc2nnnn2n1 C1(CNC(c2cc(CC)n(C)n2)=O)CC(C)(C)CN1C(=O)CC(O)CCSC c1(C2N(C(c3ccc(-c4nnc(C)s4)s3)=O)CC2)ccc(-c2cn(CO)nn2)cc1 C(=O)(CC(C)(O)C(F)(F)F)NCCCNC(=O)NC1CC(C)(C)CC(O)C1 C(=O)(CCCS(N)(=O)=O)N1CC(C)(C)C(CNC(C2CCn3ccnc3C2)=O)C1 Cc1cc(NC(=O)C(C)C)sc1C(N1CC(CNC(c2ccc(Cl)cc2)=O)C1)=O c1(OC)ccc(CCC(=O)N(CCCN(C)C(C2(C(F)F)CCCO2)=O)C)cc1 CCCC(CCC)C(=O)NC1COCCN(Cc2ccccc2I)C1 c1(C(N2CCCC(N(C)C(C3CC(C(F)F)C3)=O)C2)=O)nccc2ncncc12 c1(C(N2C(CNC(Cc3n(C)ncc3)=O)C3CCC2C3)=O)nc[nH]c2nccc1-2 N1(C(CC2C(NC(C3C(CC)OCC3)=O)CCC2)=O)CCc2ccc(C)cc21 CC1CC(C(=O)NCCc2ccsc2)CN(C(=O)C=Cc2ccn(C)c2)C1 C1(OC)(CNC(c2ccn(C)c2)=O)CN(C(=O)Cc2scnc2C)C1 c1(OCCNC(=O)NC2CCN(CC(CC)O)CC2)cccc(OC)c1 S(=O)(=O)(c1c2c(nn1C)CCC2)N1CCCC(Cc2cccc(C)c2)C1 N1(C(c2c(F)cncc2Cl)=O)CCC2(CCCN2c2nc3ncc(Cl)cc3o2)C1 c1(C(=O)OC)cc(C(C)=O)c(NC(C2CC(NC(c3ccc(I)cc3)=O)C2)=O)[nH]1 c1(CNC(C(C)OCOC)=O)ccccc1CNC(C1CC(=C2CC2)C1)=O C(C)(C)(CC(=O)N(C1CCN(C(=O)CCCCC2CC2)C1)CCO)OC N1(C(COCCC(C)C)=O)CC(CNC(=O)C=Cc2ccoc2)C(C)(C)C1 c1(C(=O)NCCCC(C)NC(CSCCOC)=O)nnccc1C c1(C(C)F)ccc(C(N2CC(CNC(=O)C(C)Cc3ccccc3F)C2)=O)cc1 C1(CC=C)(NC(=O)C(C)C(O)CC)CCCN(C(=O)C(c2cccc(F)c2)C)C1 C(=O)(C(F)CC(C)C)NCCCC1N(C(CCn2ccc(C)n2)=O)CCC1 c1(-n2cc(C3CN(C(C4CC(CC)C4)=O)CC3O)nn2)cc(F)cc(F)c1 c1(C(N2CC(C)(NC(C=CC=CC)=O)C2)=O)cnc2c(c1)N(C)CCO2 CN(C)NC(=O)CCC(=O)N1CC(NC(=O)C(C(C)(C)C)N2CCCC2)C(O)C1 N1(C(CNS(CCOCC)(=O)=O)=O)CC2(C1)CN(C(=O)CN1CCCC1CO)C2 c1(CC(=O)NCC(CN(C(C(C)(CO)OC)=O)C)C)cc(Cl)cc2c1OCC2 C1(CCOCC(=O)NCCN(C2CCCC2)CC)CCC(C)O1.C1CS1 c1(C(C(=O)NC2CC(F)(F)C2)N(CCC#C)C2CC2)cc(F)ccn1 C1(CNC(C2(SC)CC2)=O)(CNC(C2(C)C=CCCC2)=O)CCCCC1 C1(C(=O)NC(CCC)C)CCN(C(=O)Cc2cncc(O)c2)C1(C)C n1(COCC)nnc(C(N2CCC(N(C(=O)CC34CC(C3)C4)CC)CC2)=O)c1N Cc1c(Cl)c(C(=O)NCC2CN(C(=O)CNC=O)C3CC23)nn1C C=CCCCCCC(=O)Nc1cccc(NC(=O)Cc2ncsc2Cl)c1 C(=O)(C1=NOC(C)C1)NC(C)CN(C(=O)CC(C)NC(C1CCCCC1)=O)C Cc1nc(C)c(C(=O)N(CC(C)C(=O)Nc2c(C)noc2C)C)o1 N1(C(C#CC(OCC)OCC)=O)CCC2(CC1)CN(C(c1sc(O)nc1C)=O)C2 c1(C(=O)NC2CCC(NC(Cc3cn(CC)nc3)=O)CC2)ccc2cc[nH]c2c1 CCC(CCC(=O)N1CC(N(C)C)C(C)C1)NC(c1ccsc1Cl)=O c1(C(=O)NCC2CN(C(C3CC(O)C3)=O)CC23CC3)ccc2c(c1)CCCO2 c1(C(=O)NCC2CC(C)N(C(C3CCCC(C)CC3)=O)C2)ccc2cc[nH]c2n1 C1(C2CC2)(C(N2C(CNC(C3CC3C3CCC3)=O)CC2)=O)CCOCC1 c1(C(N2CCC(NC(c3cn4ccnc4s3)=O)C2)=O)cc2n(n1)CCCNC2=O c1(COC)ccc(C(=O)OCC2CC(C(F)(F)F)CN2C(=O)OC(C)(C)C)cc1 CC1(C)CCCN(C(=O)C2=COCC2)C1CNC(=O)CC1CC(=O)NC(=O)C1 c1(CNC(C(COCC)n2cc(CSCC)nn2)=O)cc(C)ccc1OCC N1(C(C(C)SC(C)C)=O)CCC(N(C)C(c2ccc(C(=O)C3CC3)cc2)=O)CC1 N1(C(C=Cc2nc(C)sc2)=O)CC2CCC1C(CNC(=O)C1=CCCCC1)C2 Cc1cccc(C(F)C(=O)NCCCCCN(C(=O)Cc2ccsc2)C)c1 CC(O)(CC(=O)NC12CCC(C(=O)Nc3ccc(C4CC4)s3)(CC1)C2)CC(=O)O CC1CC(NC(=O)CN(c2ccccc2)C)CCN1C(=O)CC1CCC1 N1(C(c2cc(C)c(CO)cn2)=O)CC2(CCN(C(C3CCCC(O)C3)=O)CC2)C1 C1(C)(C(=O)NCC(C2CCN(C(C3(O)COC3)=O)CC2)(C)O)CCCNS1(=O)=O Cc1nc(CCNC(N2CCC(CN3CCOCC3)C2)=O)cs1 C1(CC)(NC(c2ccc(O)c(CO)c2)=O)CCN(C(=O)Cc2ccccn2)CC1 O=C1CCCC(CCCC(=O)N2CC(C3CN(C(C4CC4(F)F)=O)CCO3)C2)N1 c1(-c2c(OC)cccc2)ccc2cc(C(=O)Nc3ccnc(OC)c3Br)sc2c1 C1(C(=O)NCC(C(C)C)C)(CNC(=O)C=CC2CCC2)CC12CCC2 CCCCC(C(=O)NC1CC(CN(C(=O)COC2CCOC2)C)C1)N(C)C c1(C2CCN(CC(C)(C)C#N)C2)ccccc1Br C12(C(=O)NC3CN(C(C(C(CC)C)c4ccccc4)=O)C3)CCC(O)(CC1)CC2 C(=O)(CCC(=O)C(C)(C)C)N1CC=C(C(=O)NCC(C(C)O)C)CC1 c1(C(N2CCC(C(C)(C)NC(C3OCCN(CC)C3)=O)C2)=O)cc2scnc2[nH]1 N1(C(c2sc(C3CC3)nc2Br)C(=O)NCCCSC)CCOCCC1C(C)C N1(C(Cc2c(C#C)cccc2)=O)CC2(CCC2)CC1CNC(=O)C(C)(C)OCC C1(CNC(C(CC)Sc2ccccc2)=O)CCN(C(C2CSCN2C)=O)CC1C C(=O)(CS(=O)(=O)C(C)C)NCCCC1N(C(CCC=C(C)C)=O)CCCC1 C#CCC(CC(F)F)C(=O)N(CCNC(=O)CC1Cc2ccccc2O1)CC C1(CNC(c2c(C(C)C)ocn2)=O)CC2(CO1)CN(C(=O)C(C)C#N)C2 Cc1c(C(=O)NC(C)CN(C(=O)C2=NNC(=O)CC2)C)ccc(C(F)(F)F)c1F c1(C(=O)NCCCC(C)NC(c2cc(OC)c(Cl)cc2)=O)c(F)ccc(F)c1N C1(C(=O)NC2(C)CCN(C(c3scc(OC)c3)=O)C2)CCC(C2CCCO2)O1 C1(C(N2CC3(CN(C(C)=O)C3)C2)=O)CC2(CCN(C(=O)COC(C)=O)C2)C1 c1(NC(C(C)N(CCC)C(c2ccc(C)nn2)=O)=O)ccc2nc[nH]c2c1 Cc1cc(C(=O)NC2CC(F)(CNC(=O)CC(O)C(C)C)C2)cc(O)c1 c1(C(=O)NCCCOCCN(C(Cn2c(C(C)C)nnn2)=O)C)ncncc1Cl N1(C(c2[nH]cc(CC)c2)=O)CCC2(CC(NC(=O)CSc3ccncc3)C2)C1 CCC(CCC(=O)N1CC(OC)C(F)C1)OC.C12(CC(CO)C1)C(=O)N2 C1(CNC(C(C)NC(N)=O)=O)CCC2(CCN(C(c3ccoc3)=O)CC2)CO1 C(C)(C(O)C(=O)NCC1(NC(=O)C(C)(C)OC(C)C)CCOCC1)SC c1(OC)ccnc(NCCC(C)NC(=O)C(C2CCCCC2)C)n1 C(=O)(C(C)(C)CNC(=NC)NCCc1nc(C(F)(F)F)no1)OC Cc1cnc2c(cnn2CC(N2CC(CCNn3ccnc3)C2)=O)c1 Cc1cc(C(=O)N(C2CCN(C(c3sccc3C)=O)CC2)CCO)[nH]c1C C(=O)(C1(C)CCc2ccc(Br)cc21)N1CC(C2CN(C(=O)OC(C)(C)C)C2)C1 N1(C(C2(CC)CCNC2=O)=O)CCCC(CCNC(c2ccc(C)nc2)=O)CC1 c1(C(N2CCC(C)(CNC(C(C(C)C)C)=O)CC2)=O)ccc2cc(O)ccc2n1 N1(C(C2(C)CC(=C)C2)=O)CC2CCC(N(C(=O)CSc3ccncc3)C)C2C1 C1(CCCNC(Cc2nc(C)oc2)=O)CN(C(c2cnc(C(N)=O)s2)=O)CCO1 CC1CCN(C(=O)Cc2sccc2Cl)CCN1C(=O)C(O)CC(F)(F)F CC1CN(C(c2cnsn2)=O)CC1CNC(=O)C(C)(C)CF Cc1nn(C)c(C(N2CC(CNC(C3CC3F)=O)C(C)C2)=O)c1Cl C1(C(N2C(C)CN(C(c3cc(Cl)ns3)=O)CCC2)=O)CCc2ccccc2CC1 c1(C(N2CCC(OCCNC(C(F)OC)=O)C2)=O)ccc(C)c(C(F)(F)F)c1 C1(CC)C(C(N2CC(CNC(=O)C(N3CCCCC3)C)C2)=O)CCN1C Cc1ncc(C(N2CCC(CO)(NC(=O)C3CC3)C2)=O)cc1C(F)(F)F C(=O)(CCC=CBr)NC(CN(C(=O)C(C)(C)c1ccc(Cl)s1)CC)C CCCCC(C(=O)NC(C)(CNC(=O)Cc1ccn(CC)n1)CC(C)C)N(C)C CC(C)(C)CCCC(=O)N1CCCCC(C(=O)NC(C)(C)C(C)(C)C)C1 Cc1cccc(NC(=O)C(N2CC(n3cc(C(C)O)nn3)C(C)C2)=O)c1 c1(C(=O)NC(CNC(C(C2CC2)OC)=O)CC(C)C)cc2scnc2[nH]1 Cc1nn(CC(F)F)cc1C(=O)NC(C)(C)CCNC(C1COC(C)C1)=O N1(C(CC=C=C)=O)CCC2CCCC12CNC(=O)C=Cc1cnc(C)nc1O C1(N(C(Cc2cn(CC)nn2)=O)C)CC2CC1N(C(C1C(C3CC3)C1(F)F)=O)C2 N1(C(C(C)OCC=C)=O)CC(N(C)C)C(CNC(=O)CCOC2COC2)C1 c1(CC(N2CC(CC)C(NC(C3CCCOC3)=O)C2)=O)c(F)cncc1Cl C(CCC(=O)NC(C1CC=CCC1)C(N1CC(C)(CC)C1)=O)OCC=C N1(C(C2(C)CC(=C)C2)=O)CCC(C2CCN(C(=O)Cn3cccn3)C2)C1 C(CC(C(=O)N1CCCCC1CF)NC(=O)Cc1ccn(C)n1)OC N1(C(C=CC(C)C)=O)CCCC2(C1)CN(C(C1CCCNS1(=O)=O)=O)CCO2 c1(NCC)c(C)noc1C(F)(F)Cl.C12(CCCC1)c1cn(nn1)CCCCN2 Cc1ccc(OC(F)F)cc1C(N1CC(c2ccccc2)C(C)C1)=O c1(OC)ccc(NC(C2C(C)CCN2C(c2ccc(N)cn2)=O)=O)cc1C S(=O)(=O)(c1cccc(Br)c1NC(c1ccc2ccccc2c1)(C)C)NC c1(C(=O)NCC2N(C(c3ccc(CCCC)cc3)=O)CCC2)cc2sccn2c1 N1(C(CCC=C)=O)CCCC1C1CCCN1C(c1cncc(Cl)c1Cl)=O c1(OC)ccc(CC(N2CC(N3CCN(C(=O)C(O)C(C)C)CC3)C2)=O)cc1Cl C1(C(=O)NCCC2CCCN(C(C3CCCN(C)C3)=O)C2)CCc2nccn2C1 C1(=CC(=O)Nc2nc(-c3cccc(CO)c3)cs2)CCN(Cn2ccnn2)CC1 c1(CCC(=O)NCC2(F)CC(C(=O)NC3C(=C)C3)C2)ccc(C(F)(F)F)c(F)c1 c1(C(=O)NC2C3CN(C(CC4C(C)(C)C4(C)C)=O)CC32)nc2cc(O)ccc2[nH]1 c1(C(N2C(CN(C(CN(C)C(N)=O)=O)C3CC3)CCC2)=O)cc(Cl)cc(Cl)c1N CC1CC(C(=O)NC2(C3CCCN3C(c3cccnc3Cl)=O)CC2)CC(C)(C)C1 Cc1c(C(=O)NC(c2nc(C(N3CCCC3CC(C)(C)C)=O)co2)C)ccn1C Cc1ncccc1C(C)NC(C1CCC(C2CC2)N1C(=O)CN1CCCCC1)=O c1(NC2CC(NC(C34CCCCC3OCC4)=O)C2)ccnc2ncnn12 N1(C(c2csc(CC3CCC3)n2)C(=O)NC)CCC(C)(CO)CC1 C=C(C)CCCC(=O)NC(C1CCOC1)CNC(C1(Cc2cnn[nH]2)CCCC1)=O c1(C(=O)NC(CC)CNC(C2CC2C(F)(F)F)=O)cc2ccccc2n1CC#N C1(NC(CCC(=O)N(C(C)C)C)=O)CC2CCC1CN(C(=O)CO)C2 c1(C(N2CCCC(NC(=O)CC3CC3(Cl)Cl)(CO)C2)=O)ccn2ccccc12 C1(C(=O)NCC2CCO2)CC(O)CN1C(c1ccnc(Cl)n1)=O C1(NC(C2OCC(C)C2)=O)CCCOC12CCN(C(=O)CSC(F)F)CC2 c1(CC(N2CC(CNC(CCCC)=O)C2)=O)c(C)[nH]c2ccnn2c1=O N1(C(C2N=C(C)SC2)=O)CC2(CCN(C(=O)CN(C)S(=O)(=O)N(C)C)C2)C1 C1(NC(c2ccccc2)=O)CN(C(c2csc(C(F)F)n2)=O)Cc2ccnn2C1 C1(CNC(c2n(CCOC)ncc2)=O)CC(F)(F)CN1C(=O)C(C1CC1)SC Cc1cc(CN2CCN(C(=O)Nc3ccc(Cl)cc3Cl)C(CO)C2)cc(C#N)c1 CCC1=NOC(C(=O)NC2CCC(NC(C3CSCC(=O)N3)=O)CC2)C1 c1(C(N(CC(C)O)CCNC(C(=O)NCC)=O)=O)cc(S(N)(=O)=O)co1 c1(C(N2CCN(Cc3cccn4ccnc34)CC2)=O)cc(Cl)cc(Cl)c1O S(=O)(=O)(CCNC(=O)CC1CC(NC(c2cnsc2C)=O)C1)NC c1(OC)ccc(NC(=O)C(N2CCOC3CC23)c2cocc2Br)c(C)c1 C1(N(C(=O)C=CBr)C)CCC(CN(C(=O)CCOC2CCC2)C2CC2)CC1 CCC(C)CC(C(=O)O)NC1CCN(C(=O)CCCc2nc(C(C)C)no2)CC1 CCC(C)C(C(=O)NC1(C)CS(=O)(=O)C1)NC(=O)C(C)CC(F)F C1(NC(CCC)Cc2ccc(F)cc2)CNC(=O)C(C)(C)C1 c1(C(N2CC(COC)(CNC(C3(C)CCCC3O)=O)C2)=O)ccc(Cl)c(F)c1F C12(CNC(C3C(C)CCCN3)=O)CCCC1C2(F)F C1(N(C(COCC(=C)C)=O)C)CCCCN(C(=O)Cc2conc2C)C1 C1(c2n(C)ccn2)NCCCC1C(=O)NC1CCN(c2ccc(F)cn2)C1 C1(C=C)(C(=O)NCc2n(CCC)ncn2)CCN(C(C2CC=C(C)CC2)=O)C1 c1(C(=O)NCCC(C)CCNC(=O)CC2(C(F)F)CC2)cc(F)ccc1F C1(NC(CCCCOC)=O)C2CCN(C(=O)Cn3ccnn3)CCC12 Cn1ncc2nc(Cl)nc(N3CCC(CNC(=O)CC4CCCCC4O)C3)c12 C(=O)(C(F)(F)C(C)(C)O)N1C(CNC(C(CC)Cc2ccccc2C)=O)CC1 N1(C(c2c(F)ccc(C)c2)=O)CC2CC(NC(=O)Cc3ncc(Cl)s3)CC2C1 N1(C(=O)OC)CCC(C)(CNC(=O)C(C)NC(c2cccs2)=O)C1 N1(C(C2ON=C(CC)C2)=O)CCC2(CC2NC(=O)CC2COCCOC2)C1 Cc1c(NC(c2cccc(Cl)c2C)C2CC2C)cccc1Cl N1(C(c2c(C)cc[nH]2)=O)CCC(CNC(=O)C(C)OCCN(C)C)C12CC2 c1(C(=O)NC(CCOC)CNC(=O)Cc2ccsn2)cc(F)cc2nc[nH]c12 C1(C2CN(C(C3(F)C4CCCCC34)=O)C2)(NC(c2nccc(C)n2)=O)CC1 CC(CC(=O)OCc1ccccc1)NCCOC1CN(C(C2CC2C)=O)C1 N1(Cc2c(C)ccc(C)c2O)CCC2(CCCC2C(=O)NC(C)(C)C)C1 C=CCC(CNC(=O)CC12CCC(CC1)C2)C(=O)NCC(C)CC1CCCC1 c1(CC)ccc(CCCC(N2CCOCC2CCNC(=O)CC(C)OC)=O)cc1 n1(CC(=O)NC(CNC(CCN(C(C)=O)C)=O)(C)C(C)C)nc(O)ccc1=O C=CCC(CC(C)C)C(=O)N1CC(C(=O)NCCCNC(C)=O)(SC)C1 N(C(=NCCCC1CC1)NC1CC1c1ccccc1)CC(c1ncn(C)c1)O C=CCC(CC)C(=O)N1CCN(C(C2(C(=O)OC)CC3(CCC3)C2)=O)CC1C c1(C(N2CC(NC(C3C(=C)C3)=O)(CO)C2)=O)cnc(C2CC2)nc1O c1(C(N2CC(CC(C)NC(C(C)OCC3CC3)=O)C2)=O)cccc2c1CCC2 C1(C(=O)NCCOCCCN(C(CC(C)SC)=O)C)CC2(CCCCO2)C1 C(C=CCN(C(=O)C=C)C)(CC)=CCC.C1(=O)CCN1 N1(C(=O)Cc2c(O)ncnc2O)CCC2(CCCN2C(=O)CCOC2CC2)CC1 C1(C(=O)NCC(C)NC(c2cn3c(n2)SCC3)=O)CC(C)(C)CC(C)(C)C1 N1(C(=O)CC2OCCO2)CCC(NC(=O)C(F)(F)c2ccccn2)C(CO)C1 C(CS(=O)(=O)CC(=O)N1CCN(C(c2cncs2)=O)CC1C1CC1)OC C(=O)(C(C)(C)C1CCCCC1)N(CCC(N)C1CC1)C(C)C c1(N(c2cnc(CC)nc2)C(=O)Nc2ncc(F)cn2)cnc2c(c1)CNCC2 CCCCC(C)(C)NC(=O)C(C)NC(=O)CC=CC1CC1 C(C)(c1cnn(C)c1)=CC(=O)N(CCC(C)NC(C1(C=C)CC1)=O)C N1(c2c(C#N)ccnn2)CC2(C1)C(NC(=O)CCn1cc(Cl)cn1)CCS2(=O)=O C=CCC(C)(C(=O)NCC(O)CNC(c1ccc(F)cc1OC(C)C)=O)N(C)C C#CCC(C(=O)OC)NC(c1cc(CNC(c2ccc(SC)o2)=O)nn1C)=O c1(OCCNC(C(=O)N(C)Cc2onc(CC)n2)=O)cccc(Cl)c1Cl C1(C(N(CCCOCC)C)=O)CCC2(CC2)N1C(=O)C(O)C1CCC1 Cc1cc(C(=O)NCCCNC(C2CCCN2C(c2ccoc2)=O)=O)nc(C)c1 C1(C(C(=O)NCC2C(NC(C(=O)NCC)=O)CC2)O)CCS(=O)(=O)CC1 C(C)(CCCCCO)NC(C1C(CC)N(C(=O)CSCCC#N)CC1)=O Cc1ccc(C(=O)NC2(C)CC(NC(C3CCOC3C)=O)C2)c(N)n1 c1(CC)c(C(N2CC(NC(C3CC(=O)N(C(C)C)C3)=O)C(F)C2)=O)csc1C c1(C(N(CCNC(CC(C)CF)=O)CCOCCO)=O)cncc2nc(O)[nH]c12 C1(C(=O)NCCCN(C(C2(C)CCNC2=O)=O)CC)CC(S(C)(=O)=O)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCC(COC)(NC(=O)C(F)CC2CCOC2)C1 N1(C(CC2OCC(C)OC2)=O)CCc2ccc(C(N3CCCC3)=O)nc2C1 CC(C)(C)CCCC(=O)NCC1CC(C)(C)CN1C(c1ccc(S(C)(=O)=O)o1)=O N1(Cc2ccc(COC)o2)CCCC(CNC(c2nc(C)sc2C)=O)C1 N1(C(c2cc(C)sn2)=O)CCC(C(C)(C)NC(c2oc(C(C)C)nc2C)=O)CC1 N(C1COCc2cccnc21)C(c1ccn(CCN)n1)=O C(=O)(C(Cn1cncn1)NC(=O)C(C1CCCCC1)=O)NC(CN(CC)CC)C CC(CCC(C)(C)C)C(=O)NC(CO)CCCCNC(c1cc(Cl)c(Cl)s1)=O N1(C(C(CCC)C#N)=O)CC(NC(c2cccc([N+](=O)[O-])c2)=O)CC(C)(C)C1 Cc1cn2c(n1)CC(C(N1C3CCC1CC(NC(=O)C(C)(C)CO)C3)=O)CC2 C1(CNC(C(F)=C(C)C)=O)CC(NC(c2cc(C(C)(C)C)no2)=O)CC1O c1(C(C)C)nc(NCCc2cccs2)cc(=NCC(F)(F)C(F)(F)Br)[nH]1 N1(C(c2ccn(C(F)F)n2)C(=O)NC(C)C)CCCCCC1c1cccc(F)c1 C(=O)(C(CCC)C(C)C)NC(CC#C)(C)C(=O)N(C1CCCC1)C C123CC(NC(C4CCCN4CC)=O)(CN1C2=O)C3.c1(COC)cccc(C)c1F CCC(CN(C)C)C(=O)NCC(C12CCC(CC1)C2)NC(c1cc[nH]c1C)=O C(=O)(C1=CCCSC1)N1CC(N(C(C(CC#C)C)=O)C)C(O)C1 CON1CCC(C(N2CCC(N(C(c3csc(=N)[nH]3)=O)CC3CC3)CC2)=O)CC1 c1(NC(C(c2ccc(Cl)cn2)N(C(CC)C)C)=O)ccc(F)cc1C c1(C(C(N2CCC(CC(=O)N(C3(CN(C)C)CC3)C)C2)=O)=O)ccc(C)cc1 N1(C(Cc2nnc(C)o2)=O)CC(C)(C)OCC1CNC(=O)C(c1cccnc1)C N1(CC2CN(Cc3nc(C)[nH]n3)C2)CCN(C(C2C3COCC23)=O)CC1 N#Cc1sc(C(=O)NCC2CC(CNC(c3cccnc3)=O)CO2)cc1Br C(=O)(C1CCCc2cncn21)NC(CN(C(COc1cccc(OC)c1)=O)C)C C1(C(=O)NCCC(C)N(C(C(=Cc2ccncc2)C)=O)C)CCCC2(CCC2)C1 CCCC(CC)CCC(=O)N(C(C)C(=O)N(CC)Cc1ccoc1)C C1(c2ccccc2)(NC(C(C)c2ccsc2)=O)CC(NC(C2CC2(F)F)=O)C1 c1(CC(=O)OCC(CC)(C)C)cc(C(F)(F)F)ccc1Br c1(OCC(=O)NCCN(C(c2cccc(CC)n2)=O)CC)ccc(Cl)cc1F CCCC(CNC(=O)C(C)(C)O)C(=O)N1CC2(CC(F)C2)C1 C1(Cl)(C(=O)NCC2C(OCC)CN(C(=O)Cc3cscn3)C2)CC12CCOCC2 CCCC(C(O)C(=O)N1CCCC(C)(C)C1C)NC(=O)CCC(C)(C)OC c1(CCC)ccccc1S(=O)(=O)NC1CCCCN(C(=O)OC(C)(C)C)C1 c1(OC)cc(C)ccc1CN1CCC(CC(=O)Nc2ccnc(C(=O)OC)c2)C1 N1(C(C23CCC(OC)C2C3)=O)CCC(NC(=O)C(C)S(C)(=O)=O)C(O)C1 C1(F)(C(N2CC(C)C(NC(=O)Cn3cccc(O)c3=O)C2)=O)C(C)(C)C1(C)C N1(C(c2cc(C)c(Br)o2)=O)CC(C)N(C(=O)C2=NOCC2)CC1C c1(C(=O)NC(CC)(C)CNC(C2CSCCS2)=O)cnn(C)c1C(F)F N1(C(C(C)NC(=O)NC)=O)C2CCC1C(N(C1CCCN(C)C1)C)C2 N1(C(c2c(C)occ2)=O)CCN(C(=O)CCC(C)(F)F)C(C2CCCC2)C1 C1(C(=O)NC(C#C)(C)C2CCOC2)CCCCN(C(c2ncn(C)c2C)=O)C1 N1(C(C2C(C)C2C)=O)CC2(CC(C(=O)Nc3csnc3C3CC3)CO2)C1 N1(C(c2c(C(=O)OCC)cn(C)n2)=O)CCN(C(c2cncn2C)=O)C2CC12 c1(C(N2CCC(N(C)C(C3(N(C)C)CCOCC3)=O)C2)=O)cnn2c1CC(F)(F)C2 C1(NC(CCc2c(C(=O)OC)c(C)[nH]c2)=O)CC(O)CN(C(c2cnsn2)=O)C1 N1(C(C2CCN(C)C2)=O)CC(CNC(c2nccnc2C2CC2)=O)CC12CCC2 C#Cc1cc(C(=O)NC(C2(O)CCC2)C)ccc1Cl C1(C(=O)NC(CC)C(F)(F)F)C2CCC1CN(C(C1(Br)CCC1)=O)C2 CCCCC(CC)CC(=O)N1C2CCC1CN(C(c1ccc(F)cc1)=O)C2 N1(Cc2c(C(F)(F)F)cco2)CCc2ccc(F)cc2C1 C1(NC(C(NOC)=O)=O)CC2CCC1CN2C(C1CCCC2(CCC2)O1)=O c1(CC)cc(C(N2CCC(C(C)NC(C3CCCCN3C)=O)CC2)=O)cc(Cl)c1 N1(C(c2c(CC=C)cccc2)=O)CC2C(NC(c3cncs3)=O)CS(=O)(=O)C2C1 C(=O)(C(C(=O)N1CCN(C(c2cc(=O)cc[nH]2)=O)CC1)C(C)(C)C)OCC C(C(CC(F)(F)F)NC(=O)COCC1CCCOC1)NC(c1c(CC)ncs1)=O N1(C(C(C)SC)=O)CCN(C(=O)CNC(c2ccc(C#N)cc2)=O)C2CCCC12 C1(C(=O)NC(CN(C(C(CC)(C)CO)=O)C)(C)C)OCC2CCCCC12 C1(C2CC2)(C(=O)NC2C(NC(=O)CCc3ccc(Cl)cc3)COC2)CCOCC1 c1(CCCOCC(=O)NC(c2cc[nH]n2)C)ccccc1 c1(C(N2CC(F)(CNC(c3ccc(CO)o3)=O)C2)=O)cc(C2CC2)ccc1Cl N(C1CN(C(=O)C2=CCCS2)CCc2ccccc21)C(c1csc(S)n1)=O CC1CCCC(C(N2CCCCC2CCNC(=O)C(C2CCOCC2)C)=O)CC1 C1(C(=O)NC2CC(F)(CNC(C(c3cnn(C)c3)OC)=O)C2)CC(C)(C)CO1 c1(COC)ccc(C(N2CC(CO)(NC(=O)C(C)NC(N)=O)C2)=O)o1 CC1CCCC(C2=NN(CC3=NOC(C)(C)C3)CC2)C1 C1(CC)C(NC(=O)CCn2nc(C)cc2C)CCN1C(=O)CNC(=O)OC C1(NCC(=O)OC(=O)CSc2cccs2)CC(NC(=O)CC(F)(F)F)C12CCC2 N1(CC2C(C(C)C)C2)CCCC(C)(C(=O)NCC2CC(=O)N(C3CCCC3)C2)C1 c1(CN2CC(SC)N(c3nccc(CC4CC4)n3)CC2)ccc([Si](C)(C)C)cc1 c1(CC(N2C3CC(CNC(C(CC#C)(C)C)=O)C(C3)C2)=O)cc2ccccc2o1 Cc1cc(C(=O)NC2CC2CF)ccc1-c1cc[nH]n1 c1(C(=O)NCCNC(=O)Cc2cc[nH]n2)ccc2c(c1)NC(=O)CS2 N1(C(Cn2c(=N)nc[nH]2)=O)CC(C2CC2C(=O)NC2CCCCCC2CO)C1 C#CCC(C)(C(=O)N(c1cnn(C)c1)CC)NC(=O)C(C)OC1CCCC1 Cc1cc(C(N2CCN(C(=O)C(O)CC(C)C)CC2c2ccccc2)=O)[nH]c1C#N C(C)(CNC(=O)CNC(c1cscn1)=O)(CC(C)C)NC(CC(CC)C1CC1)=O Cc1cccc(CC(=O)NCC(C)NC(c2conc2C(F)(F)F)=O)c1 C1(CC)(CNC(C2CCOC2CNC(=O)CC2(O)CCC2)=O)CCCCC1 N1(Cc2c(C)ccnc2)CC(C)OC(C)C1.c12ccc(cc1)CNC(=O)N2 c1(C(=O)NCC2CC2NC(C2CC(O)C2)=O)c[nH]cc(Cl)c1=O c1(C(=O)NCc2csc(-c3cccs3)n2)cccc(C2C(C)(C)C2C(=O)O)c1 c1(C(=O)NC2(CCNC(C(CC)n3cccn3)=O)CCCC2)cnccc1C CC(C)CCS(=O)(=O)c1ccc(NC(C2COCC(C)O2)=O)cc1 Cc1cc(N2CCC(NC(C3CCC(n4cccc4)CC3)=O)C2=O)n(C)n1 Cn1cc2c(C(=O)NC34CC3CN(C(c3cccc(C#N)c3)=O)C4)cccc2n1 N1(C(c2c(C)ccs2)=O)CC2CCN(C(=O)C(C)NC(C3CCC3)=O)CC(C2)C1 c1(N2CCCN(CCOC)CC2)nc(=N)[nH]c(=NC2COC(c3ccccc3)C2)[nH]1 CCC(CC(=O)N(C)Cc1ccc(N2CCSCC2)cc1)C(C)C C#Cc1cccc(C(N2CCC(F)(C(=O)N(C(CC3CC3)CO)C)C2)=O)c1 CC1C(NC(c2ccc(C(C)(C)C)cc2)=O)CCCN1C(C1CC(F)(CO)C1)=O C(=O)(CC(F)(F)C(F)F)N1CC2C(CNC(=O)CC3CC3C3CCC3)(C2)C1 CC(C)CCCCC(=O)N1CC2(CCN(C(=O)C(C)CN(C)C)C2)C1 CC1=C(C(=O)NC(C)(CNC(C2(C)COC(=O)N2)=O)CC(C)C)CCS1(=O)=O CC1(C)CC(CNC(=O)CC2CCC(O)C2)N(C(=O)CCOCC2CCC2)C1 Cc1cc(C(N2CCCOC(CCNC(=O)CCC3CC3(Cl)Cl)C2)=O)cc(O)n1 C(C(C)(C)CS(=O)(=O)NC(C)=O)N(C)CC1(OC)CCSC1 c1(C(C(=O)NC(C)CCNC(c2cnc(C3CC3)[nH]2)=O)C)ccc(Cl)cc1 C1(NC(C2(C=C)CCC2)=O)CCN(c2cc(F)ncn2)CCC1CO CCCCS(=O)(=O)CC(=O)NC1CCN(C(C2CCOC2)=O)CCC1CO C12(C(N3CC(CNC(C(C)SC)=O)C(C(F)(F)F)C3)=O)CCC(C)(CC1)CO2 C1(NC(c2c(C)cncc2F)=O)CC2(CCN(C(=O)CC3COC(=O)C3)C2)C1 c1(NC2CCC(NC(C(CSC)(C)C)=O)CC2)c(Br)cccc1[N+](=O)[O-] C(=O)(C(F)(F)C(O)CC)N1CC(OC)C(NC(=O)C(C)(O)CC(C)C)C1 N1(C(C(CC)C#N)=O)CCC(O)(C(C)NC(=O)C=Cc2cccc(CO)c2)CC1 N1(C(C2(C#C)CN(C(=O)CC3CCC(C)(C)C3)C2)=O)CC(=O)NC(=O)C1C N1(C(CC(=O)OCC)=O)CCC=C(C(=O)N2CC(C)CCC2CC)C1 CCCCC(CC)CC(=O)NC(CNC(c1ccc(F)cc1CC)=O)(CC)CC C1(NC(c2cn(CC=C)nn2)=O)C2CC1N(C(=O)C(CC)n1ccnc1)C2 c1(CC(=O)N(CCNC(=O)OC(C)(C)C)CC)ncoc1C c1(C(=O)NC(C(C)NC(C2OCCN(C(C)C)C2)=O)C)csc([N+](=O)[O-])c1 Cc1cc(=O)n(C)nc1C(=O)NCC(C)CNC(=O)C(O)P(C)(C)=O c1(CN2CC(C)(CC(=O)Nc3cn(C)nc3)C2)ccc(C(F)(F)F)c2[nH]ncc12 N1(C(COC(CC)C)=O)CC2CC(C(N3CC4CC(O)CC3C4)=O)C(C2)C1 c1(CNC(C2(OC)CC2)=O)cccc(NC(C2(O)COC2)=O)c1 C1(C(=O)NCCN(CCC)C(c2ccn(COC)n2)=O)CCc2n[nH]cc2C1 Cc1cccc(C(N2CCOCCC2C(=O)NC2CC(N3CCC3)C2)=O)c1F S(=O)(=O)(c1cc(C)cnc1NCCC(C)(C)CO)N1CCCC(CC)C1 N1(C(CCCNC(=O)OC)=O)C(C(=O)NCc2cccs2)CC2CC12 CC1(C)C(CNC(C2(F)CC3(CCC3)C2)=O)CCN1C(c1cnc(N)c(N)c1)=O CCCCC(CC)C(=O)N1CCC(NC(c2ccc(-c3cccs3)[nH]2)=O)C(O)C1 C(CCCCCC(=O)NCC1CC2(CCC2)CO1)NC(C(n1ncc(C)c1)C)=O CC1CN(C(=O)COc2cccc(C(N)=O)c2)CCC1NC(=O)CN(C)C Cc1ccc(CC(=O)NC(C)(C)CN(C)C(C2CN3CCC2C3)=O)cc1O O=C(N=c1cc[nH]c(CCCO)c1)C1CCCN(Cc2cc(Br)ccc2Cl)C1 C1(N(C)NC(C)CCCNC(=O)C(CC)Oc2ccccn2)CCCN(C)C1 c1(OC)cc(C(=O)NC2(C)CCC(NC(C3(C)CCCO3)=O)CC2)c(F)c(Cl)c1 CC1C(NC(c2ccc(F)s2)=O)CCCN1C(c1ccc(=O)n(C)n1)=O C1(CC)CC(C(=O)NCC(C2CCCN2C(=O)C=CCOC)(C)C)CC(=O)N1 C(=O)(C1CCc2ccccc21)N1CCC(CNC(CN(C)C)=O)C12CCC2 N1(C(C(c2cccc(Cl)c2)OC)=O)CC2(C1)CN(C(C1OCCO1)=O)CCO2 Cc1ccnc(NCC(C)(C2CC2)NC(=O)CCN2CCCCC2=O)n1 c1(C(=O)NCC(c2ccccc2)NC(=O)CCF)nc2cncnc2[nH]c1=O C(CCCCCC(=O)NC1(CNC(=O)CCC(=O)OC(C)C)CCCCC1C)SC N1(C(c2cc(C)nn2CCO)=O)CCC(NC(C2CC=CCO2)=O)C(CO)C1 Cc1nnc2n1CCC(C(=O)NCC(C)(C)NC(=O)C=Cc1cnccn1)C2 CCC(C)(COC)CNC(=O)CC(C)CNC(c1cc(C(N)=O)co1)=O C(=O)(C(C)C(C)(C)C)NCC(c1ccc(OC)cc1)NC(=O)Cc1nocc1C c1(C(N(C)CC2OCCN(C(COCCCCC)=O)C2)=O)ccnc(C)c1C C1(NC(c2c(CC)csc2)=O)CC2CCCC(C1)N2C(=O)C(C(C)C)N(C)C c1(OC)cccc(O)c1CN1CCC(O)C(C(=O)Nc2cccc(Br)c2O)C1 c1(CCNC(=O)C=Cc2ccoc2)ccc(CNC(C2CS(=O)(=O)C2)=O)cc1 c1(C(n2nc(CCN(C)C)nc2-c2cccc(O)n2)C)ccc(C(F)(F)F)cc1 Cc1cc(O)cc(C)c1C(N1CC(NC(=O)Cn2nccc2C)C1)=O C1(C(=O)NC2CC(CNC(C3CC(CC)(CC)C3)=O)C2)CCC(C)(C)OC1 C1(NC(c2ncn(C)c2)=O)CCN(C(=O)C(C)(C)C2CC2)CCC1CO Cc1c(C(N2CCC2CNC(=O)CCc2cn(C)cn2)=O)cccc1C#N C(=O)(CC(O)CC(C)(C)C)NC1CCC(CNC(c2c(C)ccc(OC)c2)=O)C1 c1(C(N(CC(C)CNC(=O)C(=O)NCC(F)(F)F)C)=O)ccc(C(F)(F)F)nn1 Cc1ccc(F)c(C2(C(=O)OC3CN(C(C4C5CC6C(C5)C46)=O)C3)CC2)c1.CN c1(C(N2C(CS(C)(=O)=O)CCCC2)=O)ccc2c(c1)CCC2 C1(C(N2CC(C#N)(F)C2)=O)CN(C(=O)CCCC2CCCO2)C2(CCC2)C1 c1(C(=O)NC(CNC(C2(C(C)C)CC2)=O)C(C)(C)C)ccc(N)c2cnccc12 C(=O)(C(F)(F)CC1CC1)NCCC1CC(NC(c2ccc(-c3ccco3)o2)=O)C1 CCCCCCCC1CCCC1NCC(C1CC1)N(C)C C(=O)(CC1=CCN(C(=O)CC(C)(C)COC)CC1)NCc1onc(CC)n1 C(=O)(CN=c1[nH]cnc(Cl)c1N)N1CC(C)C(c2cn(CCF)nn2)C1 c1(C(=O)NCCN(CCOC)C(C23CCCC2C3(F)F)=O)ccc(OC)cc1F c1(NC(C2CN(C(N3CCOCC3)=O)C2)=O)ncncc1-c1ccccc1F CC(C(=O)NC1CCCN(c2cnn(C)c2)C1=O)C(F)(F)F c1(CC(=O)NC(CC=C)CNC(c2cc(Br)c[nH]2)=O)coc2ccccc12 c1(C(N2CCC(CNC(C3CCCCS3)=O)C23CC3)=O)cccc2oc(O)nc12 c1(CCN2C(CNC(C3(c4ccccc4)CC3(F)F)=O)CCC2)cccc(Cl)c1 C1(C(=O)Nc2c(OC)ncc(C)c2)CN(C(=O)OC(C)(C)C)CCC1(C)C C1(NC(=O)OC(C)(C)C)CCN(C(C(Cl)(Cl)Cl)c2nnnn2C2CC2)CC1 Cc1nc(C2CC2)oc1C(=O)N(C1CCCN(C(=O)CC(=O)N(C)C)C1)CCO Cc1cc(CC(=O)NC2CC(N(C(=O)CC3CC4CCC3O4)C)C2)n(C)n1 c1(C2(CC)CC2)cncc(C(=O)NC(C)C(C)NC(C2CCCC2C(N)=O)=O)c1 c1(C(=O)NC(Cc2cn(C)nc2)CO)cc(-c2ccccn2)cc(F)c1 C1(NC(Cn2c(C)c(Cl)cn2)=O)CCN(C(=O)Cc2ccns2)C12CC2 C(=O)(C(C)(C)CCCO)N(CC(CN(C(c1ccc(C)o1)=O)C)O)C c1(-c2nc(-c3ccc(OC(C)C)cc3)nn2C2CC2)cccc2c1OC(C)(C)C2 c1(CC)nc(N2CCC2CNC(c2cc(C(F)(F)F)no2)=O)cc(C#N)n1 N1(C(C(C)=CC2CC2)=O)CC2CC(CNC(c3ccc(Br)cc3C)=O)CC1C2 CC(C)C(CCNC(=O)C=CS(C)=O)NC(=O)Cc1ccc(-n2cnnn2)cc1 c1(CC(=O)NCC(CCNC(C(C2CCC2)OC)=O)O)cnc2ccccc2c1 c1(C(N2CCCC(Cc3cccc(OC)c3)C2)=O)nc2c(s1)CC(C)CC2 C(CO)(CCCCNC(=O)C(C)(C)c1cccs1)NC(Cn1ncn(C)c1=O)=O C#Cc1ccc(C(=O)NC2CN(C(=O)CC3CC4CCC3C4)CC2(C)C)cc1 N1(C(C)=O)CCN(C(=O)C(C)=C2CC2)CC1c1nn[nH]n1 N1(C(c2ccc(C#C)cn2)=O)CCC(C(=O)NOCCOC(C)C)CC1(C)C C1(NC(CCC2CCN(C)CC2)=O)CCN(C(C2(C)CCC(=O)NC2)=O)CC1F Cc1cccc2nc(C(=O)NCC3(O)CN(C(C4COC(=O)N4)=O)C3)cn12 CCC(CC(=O)NC1(C(=O)N(CC(=O)N(CC)CC)C)CCC1)C1CC1 N1(C(=O)NCC(c2cc(OC)c(O)cc2F)O)CC(C)Sc2ccccc21 N1(C(C(CC)NC(N)=O)=O)CCCC(O)(CNC(c2ccc(CSC)o2)=O)CC1 c1(C(=O)NCC(=C)CCNC(c2ccc(Br)o2)=O)cc2c(s1)CN(C)CC2 c1(C(=O)NCCC(C)NC(c2c(C)con2)=O)cc(Cl)cc(F)c1Br n1(CC(=O)NC2C(CNC(C(C)=C(CC)C)=O)C2)ccc2ccccc12 c1(CNC(CN(C2CC2)CC)=O)ccnc(C(=O)NCC2(CO)CC(F)(F)C2)c1 c1(C(N2CC(C)C(NC(=O)C(F)(F)C(C)(C)O)CC2)=O)nc2cnccc2s1 C(N=c1[nH]cnc(Cl)c1C(C)=O)C1CCN(C(c2c(OCC)nccc2)=O)C1 CCCCC(CNC(=O)Cc1cccc(OC)n1)NC(=O)Cc1c(C)cnn1C CC1CNc2c(C(=O)NCCCCNC(C3CCC4(CCC4)OC3)=O)cnn2C1 c1(C(N2CCCC(NC(c3cncc(C#C)c3)=O)CC2)=O)ccc2ccsc2c1 N1(C(C(COC)(C)O)=O)CCC2(CC1)CCN(C(c1c(C)ccnc1Cl)=O)CC2 C1(CC(=O)N(C)CCO)CC2(CC2)CN1C(C1CN2CCC1C2)=O c1(C(=O)NC2CCC(CNC(CN(CC(C)(C)C)C)=O)C2)nc[nH]c2nccc1-2 N1(C(C(C(C)C)O)=O)CC2OCCN(C(=O)CC3CCCCO3)C2C1 c1(C(N(CC(CNC(C(C)OCC#C)=O)(C)C)C)=O)cc2ccncc2cc1F N1(C(C(C(C)C)(C)O)=O)CCC(NC(c2cnsn2)=O)C2(CCC2)C1 CC(CC(F)(F)F)C(=O)NC1CCCC1NC(c1cnc2n1CCS2)=O c12ccccc1C(=O)N(CC)C2.c1(CC(=O)OCC)cn(CC)nn1 C(CC1CCCC1)(C(=O)NCc1cccnc1)NC(c1cc(C2CC2)on1)=O N1(C(N(C2CC2)Cc2ccc(N(C)C)cc2)=O)CCC(C)(F)CC1 Cc1csc2ncc(C(=O)NC(C)(CNC(=O)CCCCc3cnn[nH]3)CO)n12 C(C(C)(C)CC(=O)NC1CCN1C(C)(C)C)N(C)C.C12CC(C1)CNC2=O c1(CC(=O)NCC2CC(O)CN2C(=O)Cc2ccccn2)cccc2c1CCC2 CN1N=C(C(=O)NC2C3CC2N(C(=O)CCn2cnccc2=O)C3)CCC1=O C=CCC(CNC(c1cc[nH]c1)=O)C(=O)N1CCN(CC)CC1 N1(C(c2cc(CC)nn2C)=O)CCCOC(CNC(=O)CC2(C)CC2(Cl)Cl)C1 C(C(CNC(c1ncc(N)cc1Cl)=O)S(C)(=O)=O)NC(C(C)(C)O)=O N1(c2ccnc(COC)n2)CCC2(CN(C(c3ncc(Cl)nc3Cl)=O)C2)C1 C#CCC(CC(F)F)C(=O)NCCOC1CN(C(C2SCCCS2)=O)C1 C1(NC(C(C(C)(F)F)(C)C)=O)CCC2(CC1)CN(C(=O)CCc1cnc[nH]1)C2 c1(CC)nn(C)c(C(F)(F)F)c1C(=O)OCCc1ccc(Cl)c(F)c1 CC(Cc1ccco1)C(=O)N1CC(c2ocnc2CNC(C2(CF)CC2)=O)C1 c1(C(=O)NC(C2(CNC(C3CCN(C)C3)=O)CC2)C)ccn(CCF)n1 CC1OCCN(C(=O)C(C)CCN(C)C)C1OC(N1CCC2(CC2)C1)=O O=C(C#CC1CC1)NCC1CCN1C(C1OCCCO1)=O c1(C(=O)NC(CN(C(c2cncc(-n3cnnn3)c2)=O)CC)C)[nH]c(O)nc1C C(=O)(C#CC1CCCOC1)N1CCC(CC=C)(NC(C2CSC2)=O)CC1 c1(C(N(CCCNC(C2(C)CC2)=O)C2CC2)=O)cncc2cnccc12 C1(C2(NC(COCCOC)=O)CC2)CCCN1C(=O)CCNC(=O)CO N1(C(C2CN(CC)C(=O)C2)=O)CCOCC(F)(CNC(=O)CC2CCCC2)C1 C(=O)(C(C)CC(F)(F)F)NC1CCC(N(C(C2CCN(C(CC)=O)C2)=O)C)CC1 C(=O)(C1=NOC2(CCN(Cc3ccc(Cl)o3)C2)C1)NCc1c(C)ccc(C)c1O C1(C)(CNC(c2c(CC)cns2)=O)CN(C(c2cc3sccc3[nH]2)=O)CC1C C1(NC(C(C(C)NC(c2ccc(CO)nc2)=O)C)=O)CCC(C)(C)CC1 c1(C(N2CC(CCNC(Cc3nc(C)oc3)=O)OCC2)=O)nn(C)c(C)c1Cl C=CCC(C)(O)C(=O)NC(C1CCCCN1C(c1ccnnc1C)=O)C n1(C(C(=O)N(C2CCCN(C(CC=CC)=O)CC2)CC)C)nc([N+](=O)[O-])cc1C C1(N(C(C(CC)F)=O)C)CCN(C(=O)CC2CCCCC2OC(C)(C)C)CC1 C=CCCCC(C(=O)NCC1CC(=C)C1)NC(c1ccc(NC)cn1)=O C(=O)(C1=CCC(F)(F)CC1)NCC1CN(C(C(C)(O)C2CCOCC2)=O)C1.CC(=O)O c1(CN2CC3(C(C(=O)Nc4c(C(=O)OC)nccn4)C3)C2)cnc(Br)c(F)c1 C1(CNC(=O)C=CCO)CC2CCC1N(C(C1CCCCC1CC(F)(F)F)=O)C2 C1(NC(CCCC(=C)C)=O)CC2CCC1CC2NC(C1(C(=O)NC2CC2)CC1)=O N1(C(c2nccc(C)c2O)=O)CCC2(CCCN2C(c2cccnc2)=O)C1 c1(C(=O)NCC(CNC(c2c(OCC)ccs2)=O)CO)sc(C)cc1Cl CCCC(CC)C(=O)NCC1CN(C(=O)CCCF)C1 C1(C(N(CCC(=O)NC2CC3CC3C2)CC#C)=O)CC12CCOCC2 N1(C(c2c(C)ccn2C)=O)CCCC2(CCN(C(=O)C(CO)C(F)(F)F)C2)C1 Cc1c(C(N2CC(N(C(=O)CC34CCC(CC3)C4)C)C2)=O)sc2ccsc12 N1(C(C(C)N2CC(NC(=O)OC(C)(C)C)C2)=O)CCc2c(O)n[nH]c2C1 C1(C(=O)NCc2n[nH]c(C)c2C)(CC)CCN(C(=O)CCCOC(C)C)CC1 C1(CNC(Cc2cn(C)nn2)=O)CCN(C(C2CCCC23CCC3)=O)C1(C)C c1(C(=O)NCC(=O)NC2(CC)CCN(C(N)=O)C2)ccc2cc(F)c(F)cc2n1 C1(NC(CCC2CCN(C(C(C)n3cccc3)=O)C2)=O)CCN(CCO)CC1 c1(C(N(CCC(C)NC(C(C=C)O)=O)C)=O)cccn2cc(C)nc12 c1(C(N(CC(C)CNC(c2coc(Cl)c2)=O)C)=O)cnc(N)c(CO)c1 n1(CC(=O)NC2CC(NC(CN3CC(C)(C)C3)=O)C2)ccc([N+](=O)[O-])n1 C1(C(=O)NC2C(C)N(C(=O)Cc3cccc(Cl)n3)CCC2)CCC2(CCC2)CO1 c1(C(=O)NCCCN(C(=O)Cc2ccon2)CCO)cccc2c1CCO2 C12(CCNC(C3(CC=C)CCOC3)=O)CCC(C1)N(C(=O)CSC)C2 C=CC(O)(C(=O)NCc1cncc(Br)c1)C(F)(F)F.C123CCC(CC1)N(C2)C3=O C1(NC(c2cscc2C(F)F)=O)CCN(c2nccc(CO)n2)CCC1CO NS(=O)(=O)c1cc(C(=O)NC2CCC(NCC3CCC3)C2)ccc1Cl c1(C(=O)NCCCOCCC(=O)N(C)CCC2OCCO2)csnc1Cl C(=O)(CCCC(=O)N1CC2CC1C2C(=O)Nc1cc(Cl)ccc1F)OC C1(NC(c2c(C#C)c[nH]n2)=O)CCN(C(=O)Cn2nccc2C)CC1CO CCC1=NOC(CC(=O)NC2CC(N(C)C(C3CC(O)CN3C(C)=O)=O)C2)C1 S(=O)(=O)(c1cccc2c1OC(C)C2)NC(C12CCCCC1C2)C C(=O)(C(F)(F)C(C)O)N1C2CC(NC(C(C)SCCCC)=O)(C2)C1 C=C(C)CC(C(=O)OC)NC(=O)CCCN(C)C(c1c[nH]nc1C(C)C)=O c1(N(CCCN2CCCC2)C)nc(NCC2CCSC2(C)C)c2c(ncn2C)n1 C1(CC=C)(NC(=O)CC(NC(=O)CSC)SC2CC2)CCCC1 c1(OC)ccc(C)cc1C(=O)NCC1CN(C(=O)CSc2ccncc2)C1 c1(C(N2C(CN(C)C(C3CCCOC3)=O)CCC2)=O)ccc(F)c(CO)c1 N1(C(C(F)=C(C)C)=O)CCOCC1CNC(C1(c2ccccc2)CCCC1)=O C#CCC(C(=O)N1CC(N(C)C2CC2)C1)NC(C1CCSCC1)=O c1(C(N(C)Cc2cn(CCCCC)nn2)=O)cc(CO)ccc1-n1cccn1 Cc1nnc(O)c(C(N2CCCC(O)(CNC(c3cnc(S)[nH]3)=O)CC2)=O)c1C C1(NC(CC(CC)O)=O)(CC)CCN(C(=O)C(c2c(Cl)cccc2Cl)C)CC1 N1(C(C2(COCC)CC2)=O)CCC2CN(C(=O)Cc3ccn(C)c3)CCC12 C1(C(=O)N(CCCC(C)(C)C)C(=O)C=CCO)CCCC(O)C1.C(C(F)(F)F)OCCS Cc1cccc(C(=O)C(=O)NC23CC2CN(C(=O)Cc2c(C)n[nH]c2C)C3)c1 C1(C(=O)NCC(C2CCCCC2)NC(c2ncn(C(C)C)n2)=O)CC12CC(O)C2 N1(Cc2cn(CC3N(C(CC4(SC)CC4)=O)CC3)nn2)CCCCCS1(=O)=O C(=O)(C(C)(C)CN(C)C(c1ccnc(NC)c1)=O)NC(C1CCOC1)C#C CN=c1nc(N2CCC(CNS(C)(=O)=O)CC2)[nH]c(=NCC(C)(C)COCC)[nH]1 c1(N(CCCO)C(c2nc(-c3ccncc3)n[nH]2)=O)ccc([N+](=O)[O-])cc1 c1(C(N2CC3CC3(CNC(C3(O)CCOC3)=O)C2)=O)cccnc1SC(F)(F)F C1(C(=O)NCC(C)(C)CNC(c2cnnc(O)c2)=O)CCCc2ccccc2C1 CCCC(CC)C(=O)N1CCN(C(c2cc(C)[nH]n2)=O)CC1CC(C)(C)C C(=O)(C(C)(F)C(=O)NC(CNC(=O)CCn1ccnn1)CC(F)(F)F)OCC c1(C(N2CC(N(C)C(c3sccc3C(F)F)=O)C2)=O)cc(S(N)(=O)=O)ccc1F N1(C(=O)OC(C)(C)C)CCC(NC(=O)COc2cccc(F)c2)c2cccnc21 N1(C(CC2CCC(C)(C)C(=O)N2)=O)CCC2C(C1)NC(=O)CN2C(=O)CNC=O N1(CC2(OC)CCSCC2)C(=O)CCN(CC2CCCCC2C2CC2)C1=O C1(N(C(C(C)c2cccs2)=O)CCO)CCN(C(=O)CC2C=NN(C)C2=O)CC1 c1(OC)ccc(C)nc1NC(C1CCC(NC(=O)C=C(C)C)CO1)=O c1(OCC)c(C(N2CCCC(CNC(C3(CO)CC=CC3)=O)C2)=O)cccc1C c1(C(=O)NC2CC(N(C(CC3CC(C)C3)=O)C)C2)ccc2cc[nH]c2c1 C(=O)(CCC(=O)N1CCCC1C1(C(=O)NCC2CC(OC)C2)CC1)NCCC Cc1ccc2c(CC(C)NCC(O)COCC(C)C)c[nH]c2c1 C1(N(C(C(COC)OC)=O)C)CC2CC1N(C(c1ccn(C(C)(C)C)n1)=O)C2 c1(C(=O)NC(C2CCN(c3nnc(C(N)=O)s3)C2)C)cccc(Cl)c1F c1(NC(C2C(NC(CC3(OC)CCC3)=O)C2)=O)cnn2cccnc12 CCN=c1[nH]c(C)c(C(=O)NC(CNC(C2CCOC2C2CC2)=O)C(C)(C)C)s1 N1(C(c2nc(CCC)oc2)=O)CC2CCC2(CNC(=O)Cc2ccc(C)cc2)C1 c1(CNC(c2cc(CSCC)on2)=O)cc2n(n1)CCN(C(=O)COC)C2 C(=O)(CC(C(F)(F)F)NC(C1(C(=O)NC)CCC1)=O)N(CC(F)F)CC Cc1nc(C)c(CC(=O)NC2CCC2CNC(c2cnc(O)s2)=O)s1 CC1(CC(N2CC(CNC(c3ccn(C(F)F)n3)=O)C2)=O)OCCO1 Cc1cccc(C(=O)N(C2(CCO)CCSCC2)C)c1Cl c1(COC)ccccc1CC(N1CCC(C)(CS(C)(=O)=O)C1)=O C(=O)(C(C)C(F)(F)F)NCC1(F)CC(CNC(c2c(C)cc(SC)o2)=O)C1 c1(C(=O)NCC2CC(NC(c3cc(Cl)ccn3)=O)C(O)C2)n[nH]c2c1CCCC2 Cc1ncnc(O)c1C(N1CCC(C)(CC2(C(=O)OC(C)(C)C)CCCO2)C1)=O N1(C(c2cn(C(COC)C)nc2C)=O)CCN(C(=O)C(F)CC)CC1CCO C(C(C)(C(C)C)NC(c1ccc(C)cn1)=O)NC(C1CC(C(=O)OC)C1)=O c1(C(N2CC(CC)C(NC(C3(C)CC=CC3)=O)CC2)=O)cc2ccccc2n1C CC(C)CC(F)(F)C(=O)NCCC(C(C)C)NC(C1(C(F)(F)F)CCCC1)=O c1(OC)ccc(CCC(=O)NC2CN(C(C3CC34CCC4)=O)C2)c(F)c1 C1(NC(C=Cc2cc(C)on2)=O)CN(C(c2ccc(C)c(C)c2)=O)CC1C#N c1(NCC)ccc2c(c1)CC(NC(=O)CCCc1nc(C)no1)C2.C1(=O)CCO1 N1(C(c2nc(CNC(C(C)n3cncn3)=O)oc2)=O)CCC(C)(CO)CC1 C1(Cl)(C(=O)NCC(C)NC(=O)CCC(N)=O)CCCCC1 c1(C(=O)NCC(C2CC2)NC(=O)Cc2cscn2)cc(O)ccc1F Cc1ccncc1C=CC(=O)NCC1CC1CNC(c1ccc(C(C)O)cc1)=O c1(C(=O)NC2C(NC(C(CCC)(C)C)=O)COC2)nn(C)cc1S(N)(=O)=O C1(NC(c2cccc(C)c2O)=O)CCCCCN(C(C23CSCC2C3)=O)C1 C1(CC(=O)NCCNC(=O)Cc2cccs2)CCCCN1C(=O)CCSCC#N c1(C(=O)NCCC2CC(CNC(C(C)N(C)CC)=O)C2)ccc(OC(F)(F)F)o1 C1(C(C)C)CN(C(c2cn(C)cn2)=O)CCN1C(c1ccc(Br)c(O)c1)=O C1(C(C)(C)NC(C=CCN(C)C)=O)CCCN1C(=O)CCn1cncn1 n1(CC(C)NC(c2csc(C3CCCCC3)c2)=O)cc(-c2cccs2)nn1 Cc1cc(CC(=O)N(C2CN(C(=O)CNC=O)CC2F)C)cc(C)c1 CC1(C)CC(CC(=O)NC2CC3(CC3)C2)CN1C(=O)CCc1cnccn1 CCCC(C)(O)CC(=O)N1CCC(C)(CCNC(c2oncc2CC)=O)C1 N1(C(Cn2ccc(C)n2)=O)CC2(CC(NC(=O)CN(S(C)(=O)=O)C)C2)C1 N1(C(CC2(C)CC2(Cl)Cl)=O)CC2CCC(C1)C2CNC(=O)CNC(=O)C1CC1 C(=O)(C(C)CC(N)=O)NCCC1(O)CN(C(CCC(C)OCC)=O)C1 C(CC(CC)C(=O)N(CCNC(C1CCCN(C(=O)C(C)(C)C)C1)=O)CC)=CC c1(C(N2C(CNC(CS(CC)=O)=O)COCC2)=O)cc(Br)ccc1SC c1(N(C(=O)CCCc2cnn[nH]2)CC)nc(C)cc(=NC(C)CNC(=O)NC)[nH]1 CC(C)CC(CC(=O)NCc1conc1C(C)C)NC(=O)Cc1cscn1 c1(C(N(CCC)C(C)C)=O)nc(C)ncc1-c1nc(C2CC23CCSCC3)no1 C(=O)(CCC(F)(F)F)NC1C2CN(C(C(CCSC)OC)=O)CC21 CC1c2ccccc2OCCN1C(=O)NC1CCN(c2ccccc2)C1 c1(C(=O)NC(C2CN(C(c3c(OC)scc3)=O)C2)C)c(C)coc1C C1(O)(CC(=O)NCCN(C(C2C(C)CC2)=O)CC)CCOC1 c1(NC(C2CC(C)N2C(c2ncoc2C2CC2)=O)=O)ccc(F)cc1 c1(OC)cc(C(N2CC(NC(=O)CCc3ncc(C)[nH]3)C(CO)C2)=O)nn1C N1(C(c2ccn(C)c2)=O)CCCCCC(NC(C2CC(=C(F)F)C2)=O)C1 C1(C=O)C2CC(=O)CC12.C1(C(=O)NCC)CCCN1C(=O)OC.N1(CC)CCN1CC c1(C(N2CCN(C(C3CCC3)=O)CC2CF)=O)ccc2sc3ccccc3c2c1 c1(C(N(CC(C)NC(=O)CC2CC2c2ccccc2)CC)=O)cnc2nccn2c1 c1(OC)ccc(C(=O)NC2CC(NC(C34CCCC3(C(N)=O)C4)=O)C2)cc1OC N1(C(C2(NC(=O)CS(C)(=O)=O)C(C)CCC2)=O)CC(CO)C(C)(C)C1 c1(C(C(=O)NCc2scc(C(=O)OC)n2)OCC2CCCO2)ccncc1 C#Cc1cccc(CC(=O)Nc2cccc(C(=O)NCCc3ncnn3C)c2)c1 c1(SC)nccc(=NC(=O)C2CC2N(C(c2ccccn2)C)Cc2c(C)nn(C)c2C)[nH]1 C(=O)(C1CCSc2ccccc21)NCC(CC)NC(=O)CS(=O)(=O)C(C)C C(CC(C(=O)N(C)Cc1ncn(C)n1)NC(C1CC2(CSC2)C1)=O)OC N1(C(CCC(CC)C)=O)CCCN(C(c2c(C)cncc2C)=O)CC1CO N1(C(CCC(C)(C)NC(c2ccc(C#C)c(C)c2)=O)=O)CCc2nnnn2CC1 CN1CCN(CC(=O)NC(C(=O)NCc2nccn2C2CC2)C2CCCO2)CC1 Cc1nnc(O)c(C(=O)NC2CN(C(c3c(C)nc(C)n3O)=O)C2)c1C C1(CNC(c2c(F)ccc(Cl)c2F)=O)CC2CC(C1)N(C(c1cc(O)cs1)=O)C2 C1(O)(C(C)NC(c2cccc(=O)o2)=O)CCN(C(c2cc[nH]c(=N)c2Cl)=O)CC1 C1(NC(c2csc(C)c2Br)=O)CCN(C(=O)Cc2cc[nH]c2)CC1O C1(C(=O)NCCc2ccn(CC)n2)(OC)CCN(C(C2OCCC2C(C)C)=O)C1 C1(C(=O)NC(C)CS(N)(=O)=O)CC(N=[N+]=[N-])CN1C(c1cc[nH]c1)=O C=C(C)CC(C(=O)N1CC(F)CC1C(=O)NC1CC1c1ccnc(O)c1)OC N#Cc1cc(C(=O)NC(CNC(=O)C(F)(F)C(O)C2CC2)C2CC2)cc(O)c1 c1(C(N2CC(C(=O)NC3(c4ccc(O)cc4)CC3)C2)=O)c(F)cc(Br)cc1F C(=O)(C(C)(C)C(C)(C)O)N1CC2C(CNC(C(CC)C)=O)C2C1 c1(C(=O)NCC23C(CN(C(C(C)C4CCCC4)=O)C2)C3)cc(O)cc(F)c1F C(=O)(C(CNC(=O)Cn1ccnc1C)C(C)(C)C)NC(CCC)C(C)(C)C C1(C(N(C(CCNC(C(c2cccc(C)c2)F)=O)C)C)=O)CCC(F)(F)C1O c1(N2CCC(NC(C(C(CC)C)C)=O)C(F)C2)ncnc2sc(C)nc12 Cc1noc2ncc(N(c3cc(F)ncn3)C)cc12.N12CCCC1CNC(=O)C2 c1(C(=O)OC(C(=O)OC)C2CCOC2)cccc(NC(C)=O)c1 C12(NC(N(CCCC)C3CC3)=O)CCCN(C(=O)OC(C)(C)C)CC1C2 C(=O)(CC1=CCCCC1)N1CC(N(C(CC(C)c2ccncc2)=O)C)C(C)CC1 c1(C(C(=O)NCCNC(CC2N(C)CC=CC2)=O)(F)F)ccc(=O)n(C)c1 Cc1[nH]c(=NCC(O)CNC(c2nsnc2O)=O)ccc1C#N c1(C(N2CCN(C(C3C(OC)CC3)=O)C(CO)C2)=O)ccc2nccn2n1 c1(C(C)NC(=O)NC2(S(C)(=O)=O)CC2C(=O)O)cccc2cc[nH]c12 C#Cc1cccc(C(=O)OCC2CCN(C(=O)OC)C2)n1 Cc1cc(N(C)Cc2cnn(C)c2)nc(=NCc2ccc(Cl)c(F)c2F)[nH]1 CS(C)(=O)=Nc1ccc(C(N2CCN(C3CCCC4(CCC4)C3)CC2)=O)s1 c1(CC(N2C(CN(C)C(C3CC(CF)C3)=O)COCC2)=O)cccc(C#N)c1 CC1CN(C(C2(C)C=CCN2C(C2CC3(C2)CC32CC2)=O)=O)CC(C)N1C C1(CCC)CCCC1C(=O)NCCCCCNC(=O)C(C)OCC1CC1 C1(C(C)(C)C)(C(N2CCC(F)(CNC(=O)CCC3CC3(C)C)C2)=O)CCCCC1 N1(C(CC2(CNC(c3c(CC)n[nH]c3)=O)CC2)=O)CCOCC1CCO Cn1cc(C(N)=O)cc1C(N1CC(O)(CNC(=O)C(F)F)C1)=O Cn1cc(Br)nc1C(N1CCCC1CN1CCC1)C(=O)NCCCF C1(C(=O)NC2C(NC(C3(CC)CC3)=O)CCC2)CCCC(C)(C)O1 CC1(C)CCC(CCO)(NC(=O)NCCS(=O)(=O)NC2CCCC2)CC1 C1(NC(C2(CCC=C)CC2)=O)CN(C(C2OCCOC2C)=O)C2(CCC2)C1 C(=O)(CC(O)CC(C)C)NCC(CN(C(c1ccc(C(F)F)o1)=O)CC)(C)C c1(C(=O)Nc2cnc3cc(C)nn3c2)ccnc2ccc(Cl)cc12 Cc1cn2c(=O)c(C(N3C4CN(C(C5CCCC5C)=O)CC34)=O)cnc2s1 Cc1nsc(C)c1C(=O)NCC(CO)NC(c1cc(C)n(CC(F)(F)F)n1)=O c1(-c2nc(N3CC(C(C)=O)C3)sc2)ccccc1F.C1(C)(N2C(=O)CC2)CCCOC1 N1(C(c2cncc(C)n2)=O)CC(C(N2CCCC(C)CC2)=O)CC1(C)C c1(C(N2CC(C)(CNC(C3(OC)CCC3)=O)OCC2)=O)cnc2ncccc2c1 N1(C(c2scc(C)c2)=O)CCC(C(=O)NCC2(CN(C)C)CC2)CC1(C)C C1(CN)(CNC(c2cccc(CN3CCCC3)c2)=O)CCCOC1 c1(C(N2CC3CCN(C(C(CC)SC)=O)CC3C2)=O)cc2c(F)ccc(F)c2[nH]1 N1(C(c2c(C)n(C)nc2)=O)CC2(CCC2)CC1C(=O)NCC1(CO)CCCC1 C(=O)(C(C1CC1)NC(C1CC(CCO)C1)=O)NCCSCC C1(C(=O)Nc2cncnc2O)CCN(C(=O)CC2CCCCO2)CC1O C1(C(=O)NCC(CNC(c2cc(CC)no2)=O)OC)CCC(=O)N(C2CC2)C1 C1(NC(C(c2cccc(F)c2)C)=O)CC2CN(C(C3COC4COCC34)=O)CC12 C1(CCNC(C(CC=C)OC)=O)CN(C(c2cc(C)nnc2O)=O)CC(C)O1 c1(C(=O)NC(CCCOC)C(=O)N(C)Cc2noc(C)n2)c[nH]c2nccc-2c1 C(=O)(C(C)(C)c1cc[nH]n1)NCCNC(C1CN(C(C2CC2Cl)=O)C1)=O c1(C(N(C(C)C)CCNC(C2CCC(C)(C)O2)=O)=O)cc2cc(F)ccc2cn1 C(=O)(C1=CCC(F)(F)CC1)N1CCCCC(NC(Cc2c(C)ncs2)=O)C1 C(C(O)CC(F)(F)F)N1CCC(C2N(C(C3(CC)CC3)=O)CCCC2)C1 N1(C(C(N=S(C)(C)=O)=O)=O)CCC2(CC1)CN(C(c1cccnc1F)=O)C2 O=C(C1=CC2(CN(C(c3ccn4ccccc34)=O)C2)OC1)NC12CCN(CC1)C2 c1(C(N(C)CC2(O)CCN(C(C3CN(C)C(=O)N3)=O)C2)=O)cccc(Cl)c1F Cc1nc(N2CC(NC(C3CC(C)(F)C3)=O)CC3(CC3)C2)cc(C#N)n1 c1(OC)ccc(F)c(C(N2C3CC2CN(C(c2sc(Br)cc2Br)=O)C3)=O)c1 c1(C(=O)NC2(COC)CCN(C(CC(CC)C)=O)C2)nc(O)nc(O)c1F CCCN(NC(=O)C=CC(C)(C)NC(=O)OC(C)(C)C)C(C)C C1(COC)(CNC(C2(N(C)C)CC2)=O)CCN(C(=O)Cc2nc(CO)n[nH]2)CC1 N1(C(C=CC(=O)OCC)=O)CCN(C(=O)C2=NOC(C)(C)C2)C2CCC12 CON(CCC(=O)NCC1(OC(C)C)CCC1)C(=O)c1ncoc1C(C)C CC(C)C(C)(CNC(c1cccc(Cl)c1)=O)NC(=O)CC1CCOC1(C)C N1(C(C(C=C=C)C)=O)CCN(C(c2c(CC)ncnc2CC)=O)CC1CO CC1(C(=O)Nc2cccc(CNC(C3CCC4CC34)=O)c2)CC(C#N)C1 C1(NC(C2(OC)CC2)=O)CN(C(=O)C(C)NC(C)=O)C2(CCCC2)C1 C1(COC)(CNC(=O)CCCNC(N)=O)CCCN1C(=O)C(C)N(C)C CCC(CC(=O)N(CCCNC(=O)C(OC)OC)CC)CC(F)(F)F Cc1c(C(=O)NCc2cccc(SCCC(F)(F)F)n2)nnn1C.C1(=O)CN1 C1(C)(OC)CCN(C(C2C(C)CN2C(=O)CC2(O)CCCC2)=O)C1 Cc1nn(C)cc1CN(C(=O)CC1CN(C(C2(C)CC(C)C2)=O)CCO1)C N1(C(c2c(C)c(NC(=O)OC(C)(C)C)cs2)=O)CC2CCC(NC3CC3)CC2C1 C(C(O)CCNC(C1CC(Cn2ccnc2)CCN1)=O)NC(c1ccccc1)=O n1(Cc2ccco2)cc(C(C)(C)C)nn1.c12nnnn1NC(=O)C(C)NC2C1CC1 C1(CCNC(=O)CN2CCCC2)CCCN1C(=O)CSCc1ccccn1 C1(CNC(c2cnc(CCC)s2)=O)CN(C(=O)C(C)(C)CC)CCC12CCOC2 c1(C(N2C(CNC(c3ccc4nonc4c3)=O)CC2)=O)cnc2n1CCOC2 N1(c2nc(SC)nc(C)c2)CCC2(CNC(=O)C(C)CS(C)(=O)=O)CCCCC12 c1(OC)c[nH]nc1C(=O)NCC1CC(NC(=O)CC2CCOC2=O)C1 CC1CCN1CCNC1CN(C(=O)OC(C)(C)C)C1 N1(C(=O)CN(C2CC2)CC)CC(F)(CNC(CN(CCOC)C)=O)C1 C1(OC)CC(CC(=O)NCCC(C)N(C(=O)C2=CCCC2)C)C1(C)C C1(C(N(C(CCC)C)C)=O)CCN(C(=O)C(c2ccccc2)C)C(C)(C)C1 CC1CCOCC1C(N1CCCC1CN(C(c1nccnc1N)=O)C1CC1)=O N1(C(c2c(CC)nns2)=O)CCN(C(=O)CC2(CC)CCOCC2)CC1CCO c1(N2CC(CN(C(C(CC)OCC)=O)C)OCC2)cc(=O)n(C(C)C)c(O)n1 N1(C(C2C(OC)CCO2)=O)C2CCC1CC(c1ccnn1C)C2 N1(C(C2(C)CCC2)=O)CCOC(Cn2cc(-c3ccc(Cl)cc3)nn2)C1 c1(OC)cccc(C(c2nccn2C)C(=O)Cc2ccc(-c3nn[nH]n3)cc2)c1 CC1CN(C)CCC1NC(C1CCC1c1ccc(F)cc1)=O N1(C(c2c(OC)nccc2)=O)CCN(C(C2SCC=C2C)=O)CC12CCC2 c1(C(=O)NCC#CCNC(C#CC(C)C)=O)ncc(F)cc1F C1(C(=O)NC2C(C)OCCC2)CC2(CCN(C(C3(C#N)CCC3)=O)C2)C1 c1(C(=O)O)cc(S(=O)(=O)N2C3CN(S(=O)(=O)c4ccc(Br)cn4)CC23)ccc1F c1(C(N2CC(NC(CCSCCC)=O)C(CC)C2)=O)sc2nccc(C)c2c1C CC1CN(C(C2COCCN2C)=O)CC1CCNC(c1ccccn1)=O C(CC(O)C(=O)NCCCOCCN(C)C(C1CCCCS1)=O)SC C1(c2ccccc2)(CN)CCN(C(=O)NC2CC2C(F)F)C1 c1(CNC(C2N(C(c3nc(CC)oc3)=O)CC2)=O)ccc(C)c(C)c1 N1(C(C(CCCCC)F)=O)CCN(C(c2ccsn2)=O)C2CCCC2(C)C1 C1(NC(c2ccc(N(C)C)cc2)=O)COC2(C1)CN(C(C1C(F)(F)C13CC3)=O)C2 Cc1nc2ccc(O)cc2cc1C(=O)NC1CCN(C(C2CCC(=O)NC2)=O)C1 C1(OC)CC(NC(=O)CCN2CCN(C)CC2)CN(C(=O)CCCC2CCC2)C1 C1(CNC(C2(C)CC(C)C2)=O)CCCN(C(=O)COCc2cccnc2)C1 N1(C(CCNC(=O)NC)=O)CCCC(N(CCF)C(C2CC(O)CN2C)=O)C1 N1(C(c2c(C(C)NC(C3(CCOC)CC3)=O)noc2)=O)CCCC2OCCC2C1 c1(C(=O)NCC2CCC(C(=O)NCC3ON=C(C)C3)C2)cc(C#N)ccc1C Cc1nc(=N)[nH]c(C)c1C(N1CCN(C(=O)C(n2cc(Cl)cn2)C)C(CF)C1)=O c1(C(=O)NC(C2CCOC2)CNC(C2CC(OC)C2)=O)cnc(C)n1C(F)F n1(CC(N2CCC(CN(C)C(C3C(F)(F)C34CC4)=O)CC2)=O)ccc(O)nc1=O O=C(C#CC1CCOC1)NCc1nocc1C(=O)NC(C(F)(F)F)C1CC1 N1(C(CCC)=O)CCCCC1C(=O)NCC(CO)NC(=O)CCc1ncc[nH]1 C(=O)(C(=O)N=S(C)(C)=O)N(C1CCCC(NC(=O)Cn2cc(C(F)F)cn2)C1)C C1(C(=O)NC(C)CC(C)NC(c2cc(C(=O)C(C)C)c[nH]2)=O)(CC)CCOCC1 N1(CCNC(C(C)C2CC2)=O)CCCN(C(C2(C)COC(=O)C2)=O)CC1 C=CCC(Cc1ccccc1)NC(=O)N(CC(C)CCO)C N1(Cc2scc(C(=O)OC)c2)CCCC(C(=O)Nc2c(I)cnn2C)C1 c1(C(=O)NC(CCNC(C23C(CN(C(C)=O)C2)C3)=O)C)cc(O)nc(C)n1 C(C(C)(C)C(=O)NCC1CC(F)(F)CO1)NC(C1C(C(C)=O)C1(C)C)=O C1(O)(C(N2CC(C(C)NC(=O)C(F)(F)CN(C)C)OCC2)=O)CCCCCC1 C(=O)(C(c1ccoc1)NC(=O)C(C)NC=O)NCC(C1CCC1)OCC C(C(C)C(F)C(=O)N(C)CC1CC(F)C1)NC(c1c(C)scc1)=O N1(Cc2c(C)ncs2)CCC2(CC1)CC2NC(c1cc(O)cc(F)c1)=O CC1CC(C(=O)NCc2ccc3c(c2)CC3)CCN1C(=O)CN1CCC(C#N)C1 C(=O)(C(O)CC(F)(F)F)NC(C1CCCCC1)CNC(c1c(NCC)scn1)=O C1(CNC(C2COC2)=O)CN(C(=O)CC2CCS(=O)(=O)C2)CCC1(F)F Cc1nc(NC(C)(C)C)cc(N(C)CCNc2ccc(C(C)(C)C)cn2)n1 C1(CCSc2ccccc2OC)CC(F)(F)CN1C(NOCC#C)=O Cc1c(C#N)c(N2CCN(C(=O)CN3CC(=O)N(C)C3=O)CC2)nc2ccccc12 C1(NC(C(F)=CC)=O)CN(C(=O)Cc2c(Br)cnn2C)C2(CCCC2)C1 c1(C(N2CCOCC(NC(c3ccc(Br)o3)=O)C2)=O)ccc(Cl)cc1[N+](=O)[O-] c1(NC(=O)CNCC2(NC(C3CCCOC3)=O)CCCC2)occ2c1CCOC2 Cn1c(O)nc(NC2CCC3CN(C(=O)C(F)(F)C(F)F)CC23)cc1=O c1(C(CC)N(CC(C(=O)OC)n2cc(C(=O)O)cn2)C)ccccc1C N1(C(CSCCCC)=O)CCC(C)(C(=O)NC2CCCN(O)C2=O)CC1 c1(C(N2CCC(N(C(=O)Cc3ccc(CO)cc3)C)C2)=O)cnc(O)cc1O N1(C(CC(=O)NCC)=O)C2CCC1C(C)C(NC(=O)Cc1cccc(SC)c1)C2 CC(C)(C)C(C(=O)NCC(F)CNC(C1(C)CC=CC1)=O)c1ccccc1 c1(C(=O)NCC2CCC(NC(C(C(C)C)CO)=O)C2)cnc2c(c1)nnn2C c1(OC)cc(F)cc(C=CC(N2CC(C(=O)Nc3cc(F)ccc3F)C2)=O)c1 n1(CC)ncc(C(=O)NC2CC(NC(C3(C)CNC(=O)C3)=O)C(O)C2)c1Cl CC(CC(=O)NC(C)(CNC(c1coc(Br)n1)=O)C1CCC1)n1cccn1 C(CCC(=O)NCCCN1CCCC1C)(C(C)C)NC(CN(CC)CC)=O c1(N(C)CC2CN(CC)C(=O)C2)ccc2noc(-c3cccs3)c2c1 C1(NC(C=C(C)Cl)=O)C(C)CCN(C(=O)CC23CCC(CC2)C3)C1C C1(C(=O)NC2CN(C(c3c(OC)nsc3)=O)CC2SC)C2CCC3C(C2)CC13 C1(NC(C2CC(CNC(Cc3ccc(C)o3)=O)OC2)=O)CCCC1(C)C C1(C(=O)NCC(S(C)(=O)=O)CNC(c2csc(=N)[nH]2)=O)CC2(C1)CC1(CC1)C2 C(=O)(CCCCC(F)F)N1CCC(C)C1CNC(c1cccnc1OCCO)=O N1(C(C(CC)(CC)CO)=O)CC2C3CCC(C2C1)N(C(=O)C(C)(CO)OC)C3 CN1CCC(O)(CNC(C2C3CCN(C(C4(C)CC(C)(C)C4)=O)CC23)=O)CC1 C1(NC(COCCCC)=O)CCC(COC)CC1.C12(CCCCC1)CC(=O)N2 Cc1cc(C(=O)NC(CN(C)C)C(=O)NCCCC(F)(F)F)ccn1 C(=O)(C1CCc2nccn21)N(C)CC1CCN(C(C2(C)CC2)=O)C1 N1(C(CC2C(C)CCO2)=O)CCC(C(=O)NC2(C3CC3)CCOC2)=C(F)C1 C1(C(C)C)CCCC(NC(=O)C(=O)NCC2CCCCC2O)C1 N(C(=NCCCCC(F)(F)F)N1CCc2nnc(O)cc2C1)CC(C)C c1(OCC)ccc(SC(Cc2ccoc2)C(=O)NCCOCC(=O)OCC)cc1 c1(NC(N(CCCCl)CC)=O)c(C)nn2c1CN(C(=O)OC(C)(C)C)CC2 c1(NC(C(=O)NCC(C)NC(c2cn(C)c(=O)cn2)=O)C)ccc(Cl)cc1Cl S(=O)(=O)(c1ccccc1Cl)N(C1CN(C(c2c(C)cc(Cl)nc2Cl)=O)C1)C C#CCC(C)(C)C(=O)NCC1C2CN(C(=O)Cc3c(Cl)cnn3C)CC12 C(CC(O)CC(F)(F)F)NC(C(N1CCCC(CC(=O)OCC)C1)=O)=O c1(C(N(CC(C)NC(CCCCC(C)C)=O)C)=O)cnn2c1C(C)CCC2 c1(CNCc2c(-c3[nH]c(=N)sc3)c[nH]c2)noc2c1COCC2 Cc1ccc(C(C)C(N2CC=CC2CNC(=O)CCSCC(N)=O)=O)o1 c1(CC)csc(C(C(=O)NC2CCOC2)N(C(C)CC(C)C)CCOC)c1 C(=O)(C1=CCC(C)(C)CC1)N1CCC(C)C(NC(c2c(C)cns2)=O)C1C CCC(CCC(F)(F)F)(c1nnnn1C1(C)CC1)NC(C)Cn1ccnc1 c1(C(=O)NCC2(F)CC(NC(c3nc(C(C)C)sc3)=O)C2)cnn2ccccc12 CC(C)C(CC(=O)NCC1CCCN1C(=O)CC12COCC(C1)C2)c1ccon1 N1(C(COC2(C#C)COC2)=O)CCOC(C)(CNC(=O)C(C)(C)OC)C1 N1(CC)CCC(N=c2[nH]c(=NCc3cnn(CC)c3)[nH]c3ncn(C)c23)CC1C N1(C(c2cc(CCNC(C3(SC)CC3)=O)on2)=O)CCC2CC2C1 N1(C(C2C(C)(CC)C2)=O)CCN(C(C)CNC(=O)C(O)C2CCCC2)CC1 C#Cc1cc(C(N2CCN(C(C3CCC(C(N)=O)CC3)=O)C3CC23)=O)ccc1C Cc1nc(NC2CCCCC2NC(=O)CCc2ccc(O)nc2)cc(O)n1 C1(NC(C2CC3(CC(C)(C)C3)C2)=O)CCCC12CCOCC2 c12ccccc1N2C(C=C(C)C)=O.S(C(F)(F)F)CC.C(C(F)(F)F)NC Cc1ccc(C(=O)N(C2CCC(NC(c3cn(C(F)F)cn3)=O)C2)C)nn1 c1(C2CN(c3cc(N)c(Cl)c(O)n3)C2)noc2ccc(Br)cc12 C(CC(=O)NCC1CN(c2ncc(F)cn2)C1)(C(F)(F)F)N(C)CCO c1(C(=O)Nc2ccc(C(=O)OC)o2)cc(-c2cncc(C#N)c2)cc2c[nH]nc12 Cc1c[nH]cc(C(=O)NCC2CC2NC(c2cccc(C(F)(F)F)c2O)=O)c1=O N1(C(c2cnc(C)o2)=O)CCCCC(NC(=O)CC2CCC(C)C2)C1 CCC(CC(=O)NC1(CNC(C2CC3CCC(C2)C3O)=O)CCCCC1)C(F)F CCC1=NOC(C(N2CCC(C(C)(C)C(=O)NCc3ncc(CC)o3)C2)=O)C1 C1(C(N(C)CCOCCN=c2cc(C3CC3)nc[nH]2)=O)Cc2ccccc2CO1 C12(CNC(CN3CCC(C)C3)=O)CN(C(c3cc(=O)cc[nH]3)=O)CC1CCO2 c12ncccc1CO2.C(CCC(=O)NCCCCNC(=O)OC(C)(C)C)OC c1(CC(=O)NC2CCC(F)(CNC(c3n(CC)nnc3)=O)C2)coc2ccccc12 c1(NS(C)(=O)=O)cncc(C(=O)NCC2CCC(CO)O2)c1 N1(C(C(C(CC)C)O)=O)CC2(CCN(C(c3cc([N+](=O)[O-])nn3C)=O)CC2)C1 N1(C(c2nccc(OC)c2N)=O)CC2(C)CN(C(c3cocn3)=O)CC2(C)C1 C(=O)(C1=CS(=O)(=O)CCC1)N1CC(F)(CNC(C2COCCOC2)=O)C1 c1(C(=O)NCC(C2CCCCC2)NC(C(N2CC(C)C2)C)=O)noc2c1CCCC2 c1(C(N2CCC(CN(C(=O)CC34CCCC3C4)C)C2)=O)cc(F)c2[nH]nnc2c1 c1(C(C(CC)C)C)nc(CCn2cccn2)nn1-c1ccc(OC)cc1 C(=O)(C1=CCCCCC1)NC1CCC(N(C(=O)CCc2nnc(O)nc2O)C)C1 C1(NC(Cc2c(C)ocn2)=O)CC2CCCC(C1)N2C(c1nc(O)[nH]c(=O)n1)=O C1(NC(=O)C(F)(F)CC2CC2)CCN(C(C2CCCC3(CC3)C2)=O)CC1F CC(CC(=O)NCCCC(C)NC(c1ccc([N+](=O)[O-])o1)=O)P(C)(C)=O C(=O)(C(C)(C)Nc1ccccc1)NCC(C)NC(=O)C(O)Cc1cnc[nH]1 C(=O)(CN=c1nc(CCCC(=O)Nc2ccc(C(C)=O)cc2)[nH][nH]1)NC c1(NC(C23C(CN(C(c4cnco4)=O)C2)C3)=O)nc(Cl)cnc1Cl CCC(CCCC(=O)N(C1CC(=C)C1)C)NC(=O)CC1CCCCO1 N1(C(COCC=C)=O)CCCC1(C)C(=O)NC1(c2ncc[nH]2)CC1 C12(C(=O)NCC3N(C(CC4(C)CCCCC4)=O)CC3)CCCC(C1)C(=O)NC2 N1(C(c2[nH]cc(C#N)c2)=O)CC2CCC(C1)N2Cc1cccc2occc12 Cc1nc(C(=O)NCCCC2(NC(=O)C(C)CS(C)=O)CC2)c2ccnc-2[nH]1 c1(C(=O)NCC(CCCC)NC(=O)CC(C)NC(N)=O)ccnc2[nH]nnc12 N1(C(CC(=C)C)=O)CCN2C(=O)C(NC(c3ccc(CC(C)C)s3)=O)CC2C1 CC(CS(C)(=O)=O)C(=O)NC1CCN(C(C23CCCC2CCC3)=O)CC1F c1(C(N(CCC)CCNC(=O)Cc2csc(C)n2)=O)cnn2c1CN(C)CC2 C1(C(=O)NCCCC(=O)NC2CC2)CC2(CCN1C(=O)C(F)C(F)(F)F)CC2 c1(C(N2CC(NC(C34CCC(CC3)OC4)=O)CC(F)C2)=O)cc(F)cc([N+](=O)[O-])c1 C1(NC(C2N(CCC)CCC2)=O)CC(NC(c2oc(C(C)C)nc2C)=O)CC1O C1(NC(c2cc(C)ncn2)=O)CC2(C1)CC(NC(=O)CN1CCC(C)(C)C1)C2 N1(C(COC(C)(C)C)=O)CCCC(Cc2nnc(C(F)F)o2)C1 CCC(CC(=O)NC1CCCC1NC(c1cnc(N(C)C)nc1)=O)C1CCC1 c1(C(=O)NCCCN(C(=O)C2=CCCCC2C)CC)[nH]c2ccc(C)cc2c1C c1(OC)nc(C)ccc1C(=O)N(C)CCNC(c1ccc(C)c(C)n1)=O c1(CC(=O)NC2CN(C(CC(C)(C)C)=O)C3C2C3)ccc2c(c1)OCO2 CCC(COC)C(=O)NC(c1cccnc1)C(N1CCCC1C1CCOC1)=O N1(CCC)CCC(C(=O)NCC(C2CCCCN2C(C2CCSC2)=O)(C)C)CC1 C1(C(=O)NNC(=O)N(C2CC2)Cc2ccc(C)s2)(C(=O)O)CCC2CCCC12 N#CC(=O)C(CC(=O)OCCCOc1cccnc1)c1ccc(Br)cc1 c1(OCCC(c2nnnn2C2CCCC2)NCCCCC)cncc(CO)c1 C1(C(=O)NCc2nn(C)c(=O)o2)(OC)CCN(C(=O)CN2CCC(=O)CC2)C1 c1(-c2ccc(OC)cc2C)cccc(S(=O)(=O)NCCC(=O)OC)c1 n1(CCC(=O)NCC(c2ccccc2)(C)C)cc(-c2c[nH]nc2F)nn1.C1C(=O)N1 Oc1cc(F)cnc1N1CCN(c2ccc(Cl)cc2)CC1 C(c1cn(C)cn1)=CC(=O)NCC(CNC(C(Br)=C(C)C)=O)O C1(CNC(CCC=C)=O)CN(C(c2ccsc2Cl)=O)C(C)(C)C1 C1(C(C)C)CN(C(C2CC2C)=O)CCN1C(=O)CCc1c(Cl)cncc1Cl C1(CNC(c2c(CC)scc2)=O)CCC2(CN(C(c3cnn[nH]3)=O)C2)O1 C1(C(=O)NCCN2CC3CC3C2)C2CN(C(=O)CSC3(c4cc[nH]n4)CC3)CC12 c1(CC(=O)NCC2CN(C(c3n(CC=C)ccc3)=O)CC2C)ccc(C)c(O)c1 C1(C(N(C2CCN(C(CN(C)C(N)=O)=O)C2)C)=O)CC2(C1)C(F)(F)C21CCC1 C1(C(=O)NCC=CCNC(=O)C(N2CCOCC2)C)(CC)CCNC1=O c1(CC)sccc1C(=O)NCCN(C(C1CSC(C)=N1)=O)Cc1ccccc1 c1(OC)cccc(NNC(=O)Cn2c(-c3ccc(F)cc3)c(C)sc2=O)c1 N1(C(c2cc(C)[nH]n2)=O)CC(C(=O)N(C(C)C(C)(C)C)C)C2(CCC2)C1 C(=O)(CCC(CC)NC(C1(CO)CCCO1)=O)NCC(CCC)O c1(C(N(C2CCN(C(c3ocnc3C3CC3)=O)CC2)C)=O)onc2ccccc12 CC1=C(C(=O)N(C(C)C(=O)NC23CCC(CC2)C3(C)C)CCO)SCCO1 c1(C(=O)NC2C3(CN(C(C4N=C(C)SC4)=O)C3)CCC2)ccc2cc(C)cn2c1 N1(C(C2=C(C)OCC2)=O)CC2CC(C1)CN(C(=O)C(c1c(F)cccc1F)C)C2 Cn1cnc(C(N2CCCCCC2C(=O)Nc2cccnc2)=O)cc1=O Cc1c(Cl)sc(Cl)c1C(N1C(CNC(=O)C(C)CN(C)C)CC2CC12)=O N1(C(C(C)OCC)=O)CC2C(NC(c3ccc(N4CCC(C)CC4)nc3)=O)C2C1 c1(C(=O)NCC(CCOC)NC(c2c(C)ncn2O)=O)coc2c1CS(=O)(=O)C2 c1(C(C(=O)NCCC(C)N(C(=O)Cc2cnco2)C)O)ccccc1C(F)(F)F c1(-c2nnc(N3CCOC(C)C3)n2CCN(C)CC2CC2)cnc(O)nc1O C=CCC(CC(C)C)C(=O)NCCn1cc(C(=O)NC2CC2CC(C)(C)C)nn1 c1(OC)ccc(S(=O)(=O)N2CCC(F)(F)C(C(=O)NC(C)(C)CO)C2)c(F)c1 c1(C(C)C)nnc(C(N2CCCC2CN(C(=O)CC2CS(=O)(=O)C2)C)=O)s1 c1(C(=O)NC2C(NC(CCCOC)=O)COC2)cc2nc[nH]c2cc1N CCC(C)C(C)(O)CNC(=O)C(Cc1cc[nH]n1)NC(=O)C(C)c1cccs1 CC1(C)CC(C(=O)NC2CN(C(=O)CC(=O)NCC3CC3)CC2(C)C)C(C)(C)O1 c1(OC)cncc(C(N2CC(F)(CNC(=O)C=CCN3CCCCC3)C2)=O)n1 CC(C)(C)CC(O)C(=O)N1CCN(C(=O)CC2CCC2)CC(O)C1 c1(C(=O)NC2CCC(NC(c3nccc(OC)c3)=O)C2)c(OC)ccc(Cl)c1F C1(NC(C(C)Oc2ccccc2Cl)=O)CN(C(C2C3CCC2CC3)=O)CC12CC2 C=C(CNC(=O)C(=O)NC(c1ncn(C)n1)C)c1cccc(F)c1 C=CC(C)(O)CC(=O)NC1CC(OCC(=O)NC2(C)CC=CC2)C1 N1(CC(=O)NC(C(C)NC(C(=Cc2cccs2)C)=O)CO)CCC(C)CC1 N1(C(CCCOC(C)=O)=O)CC2(CC(NC(=O)C3CC3)CO2)C1 c1(C(N2CC(OC)(CNC(c3cc(F)cnc3Cl)=O)C2)=O)ccc(Cl)c(C)c1N N1(C(c2cnc(C(C)C)o2)=O)CCC(C)(C(=O)NCC2CC(F)(F)CO2)C1 C1(C(NC[Si](C)(C)C)=O)CC2CCCC2N1C(c1ncc2ccccn12)=O N1(C(c2ccc(Br)c(C)c2)C(=O)NCC)CCCC1(C)P(C)(C)=O N1(C(C=C=C(C)C)=O)CCC2CCCC12C(=O)NC(C1CCCC1)C C1(NC(c2c(C)nc3ccccn32)=O)CCOC12CCN(C(=O)CC(C)O)CC2 c1(OCC)cc(C(=O)NC(C2CCCN2C(C2CSC2)=O)C)ccc1C c1(C(=O)NC2CCCCC2CNC(C2CC(C(F)(F)F)C2)=O)c(F)ccc(Cl)c1F Cn1ncc(C(=O)NC2CCOCC2NC(C2CC3(CSC3)C2)=O)c1C(F)(F)F Cc1[nH]c(=NCC2CN(C(=O)COC(F)F)CCC2CO)c(Cl)cc1[N+](=O)[O-] N1(C(CCC=C)=O)CCCCC1C(C)NC(=O)CCc1ccco1 CCC(C)C(O)C(=O)N(C)CCN(C)C(c1cc2ccsc2[nH]1)=O N1(C(=O)Nc2cn(CC=C)nc2)CCC(CNC(C)=O)CC1 C1(C(N(C(CC)C(=O)NCC(C)(CC)CO)C)=O)C2C3CCC(C3)C12 C(=O)(CC(C)C(=O)NCC12CC1CN(C(=O)C1=CCCCC1)C2)OCC c1(C(N(CCn2cc(CO)nn2)CC)=O)cccc(SCCCO)n1 C1(CC(=O)NCC(C2CCCC2)NC(C2CCCC2)=O)COCCO1 CCC(CC)C(O)CNC(c1cc(CCNC(C2CCCC(=O)C2)=O)on1)=O C=C(C)CC(C(=O)NCc1ccsc1C(=O)NC(C)Cc1cnc[nH]1)OC C(CNC(C12CSCC1C2)=O)(C(=O)N1CCCC1C1CCOC1)OC N1(C(C2C(C)OCCC2)=O)CCc2nc(CNC(c3cnn[nH]3)=O)sc2C1 C(C(CC(C)C)NC(=O)C(F)(F)c1csc(C)c1)NC(c1c(CC)nc[nH]1)=O c1(CCC(=O)N(CC(=O)OC)CC#C)cc(N2CC(NC(C)=O)C2)nc(C)n1 c1(CC)cc(C(=O)N(C2(CC(=O)NC(CC)C(=O)OC)CC2)C)n(C)n1 N1(C(C=Cc2ccc(C)o2)=O)CCC(NC(=O)Cc2cccc(Cl)c2)C(C)(C)C1 C1(C(=O)OCC(c2c(F)cccc2F)=O)CCc2ncsc2C1 C(=O)(CC(=O)N(CC(O)CN(C)C(c1cc(F)c[nH]1)=O)C)NCC C1(NC(C(C)(C)F)=O)Cc2ccccc2N(C(c2ccc(C(N)=O)s2)=O)C1 c1(C(=O)NC(c2ccccc2)CNC(C(C=CCCC)O)=O)c(C)coc1CC N1(C(CC)=O)CC(NC(=O)C(c2cccc(Cl)c2)C)C2CC2C1 N1(C(C2(C)COC2)=O)CCC2(CC(NC(c3cnc(C4CCCO4)s3)=O)C2)C1 C(N=c1cc(NCc2nccn2C(F)F)nc[nH]1)C1C(CC)C1 Cc1cc(C#N)ccc1C(=O)NCc1ccc(C(N2CC(C)CC(C)C2)=O)nc1 C(=O)(CCCCC(C)=O)N1C(C(N(CCCCC)C(C)C)=O)CCC12CC2 c1(CC(N2CCC(CNC(=O)CC3CCOC3)C2)=O)ccc(Br)c(Cl)c1 C(=O)(C(C)(C)C(C)(C)O)N(C(C1CCCCC1)CSc1ccccc1)C(C)=O c1(N2CCC(C)(NC(c3ncc(OC(C)C)nc3)=O)CC2)nc(C)cc(C#N)n1 CC1C2CCC(C2)C1C(=O)NCC1(C(N2CCCCC2CO)=O)CC1 C1(C(N2CC(O)(C(C)NC(c3nccnc3N)=O)C2)=O)CC2CCCC12 C1(CC=C)(NC(C2CC3CC2C2CC32)=O)CCN(C(=O)COC(C)=O)CC1 N1(C(C(C=C=C)C)=O)CCn2nc(CNC(=O)CCNC(N)=O)cc2C1 c1(C(=O)NCc2c(CCNC(c3cc[nH]c3C3CC3)=O)ocn2)ncncc1F C(CC(C)C)(C(=O)NC(CO)C(C)NC(c1ocnc1C1CC1)=O)NC(=O)OC Cc1c(F)cc(NC(C2CC(F)CN2C(=O)Cc2cc(Br)ccc2Cl)=O)cc1Br CC(C)C(CCN(C(=O)CC(C)n1cccn1)C)NC(=O)CCCc1cnn[nH]1 C1(CC)CCN(C(c2c[nH]c(C(N)=O)c2)=O)C1CNC(c1cccnc1)=O C=C(C)c1ccccc1NC(C1CCN(c2ccnc3ccnn23)C1)=O C1(CC)(NC(=O)C(C)Cc2cccc(F)c2)CCCN(C(=O)C(C)(C)C(C)C)C1 CCCCCC(F)C(=O)N(C(C)C(=O)NCC1CCCC2(CC2)C1)CCC CC1(C)CCCC(C(N2CCC(F)(CNC(C3CS(=O)(=O)C3)=O)CC2)=O)C1 C(=O)(CCC(=O)c1cc(Cl)sc1Cl)N1CC(NC(C2(CC#C)CC2)=O)C1 C(=O)(C(F)CC(CC)CC)NCCCN(C(C(=O)OC)C(F)(F)F)C1CC1 N1(CC2C(C)CCC2)C(=O)N(Cc2nn(C)cc2Cl)C1=O N1(C(c2c(C)cco2)=O)CCC(C2CCCN(C(C3CS(=O)(=O)C3)=O)C2)C1 C(=O)(C1CCc2cccc(OC)c21)NCC1CC(NC(C(CC)N(C)C)=O)C1 c1(C(N2CC(NC(CC(C)N3CCCC3=O)=O)(CO)C2)=O)cccc2c1OCC2 c1(C2C(C)C2C(=O)NC(C)CCNC(=O)CC2(N3CCCC3)CC2)ccccc1 N1(C(C=Cc2c(C)cncc2)=O)CC(NC(=O)Cc2nocc2C)C2(CCC2)C1 c1(C(N2CCC(NC(C(CC=CC)C)=O)(CO)C2)=O)cccc2c1CC(C)(C)C2 CC(CC(=O)NOCC(=O)NC1(CCCCO)CC1)NC(N)=O Cc1nc(C(=O)NCC(C2(O)CCSC2)(C)C)sc1C Cn1cc(Cl)cc1CNC(C12CC(C1)C(C1CCN(C(=O)OC(C)(C)C)CC1)O2)=O C(=O)(CC(C)(C)CNC(C1(C)CCCCC1C)=O)N(C)Cc1n(CC)cnn1 N1(C(C2C3(CCN(C(c4cnc(=N)[nH]c4)=O)C3)C2)=O)CCCC2(CC1)CC2 c12ccc(cc1)c(=O)o2.C(=O)(C1=CCC1C[Si](C)(C)C)NC C1(CNC(c2cc(CCC)on2)=O)CCN(C(c2onc(CC)c2C)=O)CC1O CCCC(C(=O)N1CC2(C1)CC(=O)N2)NC(=O)OC.C(CC(C(C)C)OC)SC C1(C(N(C)CC)=O)CN(C(c2ccc(F)cc2I)=O)CC12CCC2 C(C(CC(C)C)C(=O)NC1(CO)CC2CCC1C2)NC(c1n(CC)nc(C)c1)=O Cc1cc(NCC(C2CC2)NC(C2COCCN2C)=O)n2ncnc2n1 Cc1[nH]nc(Cl)c1C(=O)NCC1C2CC1N(C(c1cnc(C(C)(C)C)s1)=O)C2 c1(C(N(CC)CC)=O)n[nH]c2cc(C(=O)NC3CC4OCCC34)ccc12 c1(C(N2CC(NC(C(CC#C)C)=O)CC2(C)C)=O)cc2cc(C)ccc2[nH]1 c1(CCC)ccc(CCCC(=O)NCC(C)CNC(=O)CC2CCN(C)C2)cc1 c1(SC)nnsc1NCCC(Cc1cccs1)NC(=O)OC(C)(C)C Cc1ccnc(C(=O)NCC(C)CNC(C2CC3CCC2O3)=O)c1Br c1(C(CNC(C(C2CCOC2)OCC)=O)C)ccc(F)c(F)c1 C1(NC(Cc2c(C)occ2)=O)CN(C(=O)C(C(C)C)NC(N)=O)CCC1C c1(CN2C(C)(C(=O)Nc3n[nH]c(Cc4ccccc4)n3)CC2)cc(Br)ccc1O N1(C(C2N(C)CCN(C(c3c(C)cc(F)cc3)=O)C2)=O)CC2CC(C)(C)C2C1 C1(C(=O)NCC(C)(C2CC2)NC(C2CCSCC2)=O)OC2CCC1C2 CC1CN(c2ccc(NC(C)(CCC#N)c3ccccc3)cn2)CC(C)O1 c1(OCC=C)c(C(=O)NC2CCN(C(=O)CC(C)(C)OC)CC2C)cccc1C N1(C(C=CC=CC)=O)CC(CNC(=O)C=Cc2cccc(CO)c2)CC12CCC2 CN1CCN(C(C2CCCN2C(=O)CCC(=O)C2CC2)=O)CC1 c1(C(=O)NCC2CCN(C(c3cn(C(C)C)nn3)=O)C2)ccc(Cl)c(O)c1 C(=O)(CC(C)(C)CN(C)C)N1C(CCCNC(C(COC)(C)C)=O)CCC1 c1(C(=O)NCC(C)NC(C(CCC)CC)=O)snc2ccc(Br)cc12 CC1CCN(C(c2cnc(C3CC3)[nH]c2=N)=O)CC1NC(C1(C2CC2)CC1)=O CCC(CC)CCC(=O)N(CC(C)CNC(c1ccc(Cl)c(F)c1F)=O)C C1(C(F)(F)F)(N(C)CC2OCCC2(C)C)CC2CCC1C2 Cc1ccc(CC(=O)NC(C2CCCN2C(=O)C(C)n2cccc2)C)c(Cl)n1 c1(C(=O)NCc2cccc(NC(C(C)OCCC#C)=O)c2)cc2cn[nH]c2cn1 CC1CN(C(c2cncc(F)c2)=O)CC1N(C)C(C1CCC(N(C)C)C1)=O Cc1cccc2c1CCOC2C(=O)NC(CCNC(C1(CO)CCC1)=O)C(C)C c1(SCCC(=O)NC(CC)(C)CNC(=O)C(C)SC)ccc(Cl)cc1Cl N1(C(N)=O)CCC(NC(=O)COC2CN(C(c3cc(CO)n(C)n3)=O)C2)CC1 c1(C(=O)NCC(C)NC(C2CC2C(N)=O)=O)ccc(N)c2ccncc12 c1(C(=O)NC(C2CCCN(C(=O)OCC)C2)C)cnc2cc(C)ccn12 C(CN=C(NCCF)NCc1ccccc1SC1(F)CCCCC1)OC c1(CNC(c2cc(COC)on2)c2nnnn2C)ccc(N2CCOCC2)cn1 C(CN=c1[nH]c(N2CCN(CC)C(=O)C2)nc2c1COC2)N1CCC(OCC)C1 C(=O)(C1CCCc2ccccc21)NCC(CC=C)NC(c1scnc1C(C)C)=O Cc1cccc(C(F)C(N2CCC(C)C2CNC(=O)C(C)C)=O)c1 c1(C(N(CC(C)N(C(=O)COC2(C)CCCC2)C)C)=O)ccc(N)cc1O c1(C(=O)NC(CC=C)CC(=O)N2CC=CC(O)C2)cccc(C)c1C#N N1(C(c2noc(CC)c2C)=O)CCCC(C)(NC(=O)C(N2CCC(C)C2)=O)C1 c1(C(C(N2CCC(CNC(COc3cc(C)on3)=O)C2)=O)(C)C)ccc(Cl)cc1 c1(NC(C(=O)NCC2CCN(Cc3ccccc3)C2)=O)nnc2n1CCCC2 c1(C(N(CC(CC)NC(C2C=CC=CC=C2)=O)CC)=O)cccc2ccoc12 C1(NC(c2ccccc2C(F)(F)F)=O)CCN(CC(N2C(C)CCC2C)=O)C(C)C1 c1(OC)nccc(C(N2CCC(C(=O)NCc3cc(Br)ccc3F)C2)=O)c1Cl c1(OC)ncc(F)cc1C(=O)NCC1CC1NC(=O)CC1OCCC1(C)C N1(CC(=O)NCC(CC)(C)NC(=O)C(CO)OC)CCNC(=O)C1 C(C(C(=O)NCCc1nc(CC)no1)NC(C1CC1C#N)=O)OCC CC=C=CCCN=C(NCCOCc1ccccc1)NCC1CC2CCC2C1 c1(N2CC(NC(c3cc(CCC)on3)=O)C(C)(C)C2)nc2ncc(Cl)cc2o1 C(=O)(C1=NOC(C)C1)N1CC(C#C)(C(N2CCC(C(=O)NC)C2)=O)C1 N1(C(CCN(CCOC)C)=O)CCC(NC(=O)CN2CCC(C)(C)CC2)C(F)C1 C1(c2cn(CCN(C)C)nn2)(NC(C2C(CC)CCC2)=O)CC2(CCOCC2)C1 N1(C(C=CCC)=O)CCCC(N(C(c2c[nH]nc2Cl)=O)CC2CC2)C1 N1(S(CCOCC)(=O)=O)CC(C2CCCN(C(=O)C(C)(F)F)C2)C1 N1(C(C(C(C)C)(C)O)=O)CCC2CC(CNC(=O)COCCN(C)C)CCC2C1 c1(C(N2CCN(CCOC3CC3)CC2)C(=O)NCCCC)cnn(C2CC2)c1Cl c1(C(N2CCN(C(CCC(=C)Cl)=O)C(CC)C2)=O)cc(C)c2ncccc2c1 S(=O)(=O)(c1cccc(Br)c1)N(c1c(-c2cn(C(C)C(=O)O)nn2)cccc1Cl)CC CCN(NC(=O)CCn1cc(CC)nn1)C(N)=O.N1(CCC(=O)N)CCCOC1=O C=CC(C)CC(=O)NCC1CCCC1NC(=O)Cc1sc(S)nc1C N1(C(C2N(C)CCOC2)=O)CCN(C(c2ccccc2C2CC2)=O)CC1C1CC1 C1(NC(C2C(COC)CC2)=O)CN(C(C2CCC2(C)C)=O)CC1SC C1(NC(C2(NC(=O)NC)CCCC2)=O)CN(C(c2cccn2C)=O)C2CC12 N1(C(CC(C)(C)O)=O)CC2CN(C(c3cc(C(C)(F)F)ccn3)=O)CCC12 c1(OC)nc(N2CC3C(C2)N3C(c2ccc(OC(F)F)cn2)=O)ncc1C#N C1(C#N)(C(=O)NC2C(C(=O)NCC#C)OCC2)CCCO1 c1(C(=O)NCC2(O)CN(C(C(CCC)N(C)C)=O)C2)[nH]cc2c1CCC2 C(C(C)(C)CNC(C1CCC1c1nncn1C)=O)N(C)C(C1CC(C)(C)C1)=O C(=O)(CCC(C)C)NCC(CNC(c1nc(COC)sc1)=O)(C)F C1(N)(NC(N2CCC(N(c3ccccc3)C)C2)=O)CCOCC1(C)C CC1=C(C(=O)NCC=CCNC(C2CC(Cc3cccnc3)C2)=O)CCCC1 c1(C(=O)NC2C(C(N3CCN(CCC)CC3)=O)CCCC2)ccc([N+](=O)[O-])cc1F Cc1c(C(N2CC(C)(NC(C3C4CCC(=O)C34)=O)C2)=O)oc2ccccc12 C=CC(CC)C(=O)NC1COCC1NC(=O)CCCN1C(=O)CNC1=O CCCS(=O)(=O)CC(=O)N1CCN(C(c2cn(-c3ccccc3)nn2)=O)C2CC12 C1(N(C(CN(C(C)=O)C)=O)CCF)CCCN(C(C2C3CCN2CC3)=O)C1.NC=O C(C(=O)NCCn1cncn1)(C(C)C)NC(C(F)=CCC)=O Cc1ccc(C(=O)NCC2CCCCN2C(c2cc[nH]c2)=O)c(F)c1C C1(NC(C2CC(OC)C2)=O)CCN(C(=O)Cc2cnoc2)CC(C)(C)C1 c1(CC(=O)NCC2CCCC2NC(=O)CC2(O)CCOCC2)ccc(F)c(F)c1 C(=O)(C1=COCC1)N(C(C(=O)NC(CCC)CO)(C)C1CC1)C C1(NC(CC2CCN(C(C3(COC)CC=CC3)=O)CC2)=O)CC2C(C1)C2(F)F c1(OCC(=O)N(C2CCC(CC3CCC3)CC2)C)c(F)cccc1[N+](=O)[O-] N1(C(CC=CCNC(C(C)(C)NC(C)=O)=O)=O)CCN(C)C2CC12 C1(C(N2CC(F)CC(NC(CCC#C)=O)C2)=O)CC2CCCC(C1)C2 C1(CCOC)CN(C(C2CC23CCC3)=O)CCN1C(c1cnc(COC)s1)=O CC1CCn2cc(C(=O)NC3CCN(C(C4C(C)(C)C4(C)C)=O)CC3O)nc2C1 CC1COCC(CC(=O)NCC2(C(=O)N(CCCC(C)O)C)CC=CC2)O1 CC(C)C(=O)C(=O)NC12CC(C(=O)NC3CC(F)C3)(C1)C2 C(=O)(C1CCCc2scnc21)N(CCNC(C1CCCOCC1)=O)C1CC1 CC(C)C(C)(CNC(C1(C(C)C)CCC1)=O)NC(=O)CN1CCN(C2CC2)C1=O c1(CNC(c2c(CNC(c3csc(Cl)n3)=O)n[nH]c2)=O)cccc(F)n1 c1(C(N2CCN(C(C(OC)OC)=O)C(C#N)C2)=O)ccc(Br)c2cccnc12 Nc1ccc(C(N2CCCN(C(C3CCSC3)=O)CC2CO)=O)c2ccncc12 Cn1c(C(=O)NCCOCCOCCCNC(C2(C)CC(C)(C)C2)=O)nnc1S c1(C(N2CC(NC(=O)C3=C(Cl)CCC3)CC(OC)C2)=O)cc2n(n1)CCCC2O N1(C(c2c(CC)ncs2)=O)CCC(CNC(c2cc3c(s2)CSC3)=O)C1(C)C c1(C(=O)NCC2(NC(C3CC(C)N(C)CC3)=O)CCC2)ncc2n1CCCC2 n1(CC(N2CC(CNC(C3(OC)CCCOC3)=O)C2)=O)ccc([N+](=O)[O-])n1 C1(C(N2CCC(NC(C(C)c3ccsc3)=O)C(F)C2)=O)CCN(S(N)(=O)=O)CC1 Cc1ccc(F)c2oc(C(=O)NCCOCCN(C)C(C3CCCSS3)=O)cc12 N1(C(CCCC(C)=O)=O)CC=C(C(=O)NCC2(CCO)CCCC2)CC1 c1(CNC(C(CCCC)(F)F)=O)ccc2c(c1)CN(C(c1ccoc1CC)=O)C2 N1(CC(C)C)CC(C(=O)NCC(C)(C)Cn2cc(C(C)(C)F)nn2)CC1=O c1(C(C(C)NCc2cn(CC)nn2)O)ccc(C)cc1 C(=O)(C(O)C(C)(C)C)N1CC(OCCNC(C2CCC(C(C)C)CC2)=O)C1 c1(OC)cc(C)sc1C(=O)NC(C1CCCCN1C(c1ccc(O)nc1)=O)C c1(C(=O)OCC)cc(C)n(C2CN(Cc3cc(OC)nc(OC)n3)C2)c1C N1(C(c2c(Cl)cn(CC)n2)=O)CCN(C(c2cc(N)ccc2F)=O)CC1C(C)C Cc1cc([N+](=O)[O-])cnc1C(=O)NCCCNC(=O)C(c1ccccc1)N(C)C C=CCC(C)(O)C(=O)NCC1CC1CC(N1C2CCC1COC2)=O C=C=CCCC(=O)NC(C(=O)N1CC(n2ccnc2)(CO)C1)C(C)C C(=O)(C1=CC2CCC(C1)C2)NC1C2N(C(c3ccnn(C)c3=O)=O)CC(CC2)C1 c1(N(C2CCN(C(c3c(C(C)C)cccc3)=O)C2)CCO)ncc2c(n1)CCCC2 C1(OC)CC(C(=O)NC(C)CNC(=O)C(C)(C)c2ccccc2)C1(C)C N1(C(c2n(C)ncc2Cl)=O)CCC2(CC1)OCCCC2NC(c1occc1F)=O CC(=O)CCCC(=O)N(CCCNC(c1scc(C)c1Br)=O)C c1(C(N2C3CN(C(C4CC(C)NC(=O)C4)=O)C(C3)C2)=O)cccc2c[nH]nc12 C1(C(=O)Nc2ccn(CC)n2)COC2CN(C(=O)C(c3ccccc3)=O)CC12 CC(C)C(C)(CNC(=O)CCCN(C)C)NC(c1c(C2CCC2)cnn1C)=O c1(NC(C2N(C(c3cc(CC)[nH]n3)=O)CCSC2)=O)nc(Cl)ccc1Br c1(C(=O)NC2C(NC(c3nc(C)nn3C)=O)C2)nc(C)c(C)nc1C c1(C(=O)NC2CC(CNC(C(C)SCC)=O)C2)ccc(Cl)nc1N c1(C(=O)NC(C)CNC(c2cnc(Cl)c(Cl)c2)=O)cc2c(o1)CCCNC2=O C1(C(=O)NC2(CF)CN(C(=O)NC(C)C(=O)NC)C2)CCS(=O)(=O)C1.CN C1(C(N2CC(C(C)(C)O)(CNC(C(COC)(C)C)=O)C2)=O)CC2OC(=O)OC2C1 N1(C(c2c(O)ccc(C)c2)=O)CCN(C(=O)CC2CCCN2C(C)C)CCC1C c1(N2CCCC(CC)(CO)C2)nc(N2CCSC(C)(C)C2)nc2c1CCC2 C(C[Si](C)(C)OC)C1C(C(N(C(CC)CO)CC)=O)C1 N(C1CCOc2c(C)cc(F)cc21)(C(c1cc(C2CCCC2)[nH]n1)=O)CC N1(C(C2(CCOC)CC2)=O)CCCC(C)(CNC(c2cc(Br)c[nH]2)=O)C1 N1(C(C2C(=C)CC2)=O)CC2CC(NC(c3cc[nH]c3C(C)C)=O)CC2C1 C=C(Cl)CC(C(=O)NCc1ccc(=O)n(C)c1)NC(=O)Cc1cccc(O)c1 C12(CC)COC(C(=O)NCC3CCN(C(c4c(CC(C)C)noc4C)=O)C3)(C1)C2 C1(CNC(CCCCNC(C)=O)=O)CCN(C(c2conc2C(C)C)=O)CC1C n1(CC)ncnc1C(=O)N(C)CC1CCN(C(=O)Cc2csc(C)n2)C1 C1(N(C(=O)CCNS(C)(=O)=O)C)CCCN(C(C2CC2C#N)=O)CC1 c1(C(=O)NCC2CCN2C(c2ncncc2Br)=O)cn2c(n1)COCC2 N1(C(C(CO)NC(c2cnn(CC3CC3)c2)=O)=O)CC(O)CC(O)C1 C1(N(C)C(C2OCCC2NC(c2csnc2Cl)=O)=O)CCCC1(C)O c1(C(N(CCCNC(=O)C(C2CC2)OCC)CC)=O)[nH]c2ccc(F)cc2c1Cl Cc1ccc2cc(C(=O)NC3CCCCCC3NC(c3ccc(Cl)s3)=O)cn2c1 C1(C(N2CCC(CCOC)C2)=O)(CF)CCN(C(=O)CC2CCSC2)C1 C(=O)(CC(C)C(=O)NCC12COC(CF)(C1)C2)OC.C(C)(C)(C)O c1(SCC(=O)NCC23CC(NC(C4N(C(N)=O)CCC4)=O)(C2)C3)ccccc1F N1(C(c2c(CC)ncnc2)=O)C2CCCC1CN(C(C1CN3CCN1CC3)=O)C2 c1(OCC2(C(=O)NCC(C(C)C)NC(C3C(OC)CC3)=O)CC2)cccc(F)n1 CCCC(C(=O)NC1(CCNC(=O)COCCCC(C)C)CCC1)S(N)(=O)=O c1(OC)ncccc1C(=O)NCCOCC(=O)NCc1ncn(C2CC2)n1 N1(C(C2(C)C=CCCC2)=O)CC2(CCNC(c3ccc(C(N)=O)s3)=O)CCC1C2 Cc1nc2ccccc2c(C(N2CC=CC(NC(c3[nH]cnc3C)=O)C2)=O)c1C N#Cc1cc(CNC(C2CNCCN2c2ncnc3sccc23)=O)cc(F)c1 c1(OC)ccc(Cl)c(F)c1C(=O)NC1CCC(NC(C2COCCC2(F)F)=O)C1 C1(C(=O)OC)CSCN1C(=O)Cc1cn(CC2CCCCC2)nn1 C(=O)(CC(C)C(C)C)N(C(c1c(C)nc(CNC2(n3ccnn3)CC2)s1)C)C C1(C(N(C)CC2(O)CCC2)=O)CCOC1CNC(C1(Cl)CCC1)=O c1(C(=O)NC(CNC(Cc2c(C)ccnc2)=O)C)ccc(N)cc1Cl c1(NC(C2C(=C)C2)=O)ccc(NC(C2(CCC3CCCCC3)CC2)=O)cc1C C1(C(=O)NCCCCCn2cc(COCCN(C)C)nn2)CCC(=O)CC1(C)C c1(CC)cc(N)ccc1C(=O)N(CCNC(C1(C)CC=CCO1)=O)CCOC C=C(Cl)CC(C(=O)NC(C12CC(CO1)C2)C)NC(=O)C(C)OC(C)(C)C N1(C(c2nc(-c3cn(C)nc3)oc2)=O)CC2CC(NC(c3cnc(O)o3)=O)C1C2 Cc1sc(S(N)(=O)=O)cc1C(N1CCN(C(c2cc(=O)n(C)o2)=O)C2CC12)=O Cc1cccc(CCC(=O)NCCC(C)NC(C2(O)CCOC2)=O)c1 C1(CC=C)(C(=O)NC(C)C(C)(C)OC)CN(C(=O)C(C)SC(C)C)C1 CC#CCC(C(=O)NCC(O)CC)NC(=O)CCc1cncnc1 c1(CNCC23C(CN(C(C4CCC(CO)CC4)=O)C2)C3)c(O)cccc1Cl C(=O)(C(CCOC)OC)NC1(CC)CN(C(=O)CC2(C)CC2)C1 C(CN=c1[nH]cncc1C)C1CCC(NC(C2(CCCC)CC2)=O)C1 c1(N2CCCC(NC(C(c3ccc(Br)cc3)OC)=O)C2)ncc(Br)c(O)n1 C12(C(=O)NCCN(C(c3c(NC(C)=O)cccn3)=O)C(C)C)CC(C1)C(C)(C)O2 c1(CNC(c2cc(C(=O)OC)[nH]c2)=O)ccccc1CNC(c1coc(Cl)c1)=O C1(CC(N2CC(COC)(NC(C34COCC3C4)=O)C2)=O)CCC(C)(C)O1 C1(C(C)NC(c2cscn2)=O)CCCN(CCc2ccsc2)C1 C(=O)(C(=O)N)N(CCN1C(=O)CC2CC2OCC1)CC.C(C(C)O)CC c1(C(C)C)ccc(S(=O)(=O)N2CCCC(NC(=O)C(C)(C)C)C2)cc1Cl N1(C(CC2C(OC)CC2)=O)CCC(CNC(=O)CC(=O)N(C)C)CC1 C1(CNC(c2n(CC)ccn2)=O)CN(C(=O)C=Cc2ccncc2C)CCC1C CCC(CC)CCC(=O)NCC(C1CC1)NC(c1ccc(Br)c(N)n1)=O C1(C(N(C)Cc2cn(CC3COCCO3)nn2)=O)CCCCS1(=O)=O C1(CNC(=O)CC2CC(F)C2)CCC(NC(c2occc2Cl)=O)CC1 c1(OC)ccc(CC(=O)NCC(C(C)C)NC(C2CC2c2cccs2)=O)cn1 C1(NC(C(c2cccc(OC)c2)C)=O)CCN(C(=O)CCC2CC2(C)C)CC1F c1(C(=O)NC2C(NC(C(C)OCC=C)=O)CCC2)cc([N+](=O)[O-])cc(Cl)c1Cl CC(Cc1ccccn1)C(=O)N(C)CC1(O)CN(C(=O)C(C)(C)F)C1 n1(COC)ccc(C(=O)N(C(C(=O)NCCC23CC(CO2)C3)C2CC2)C)n1 c1(CC(=O)N(C2CCC(NC(=O)C=CC3CC3)C2)C)cccc2sccc12 c1(CC(=O)NC23C(C)OC(CNC(C4CC=CC4)=O)(C2)C3)cccc2nonc12 C1(NC(c2c(CC)cco2)=O)CCCN(C(=O)CC2CCS(=O)(=O)C2)CC1 c1(C(=O)NC(CNC(C2CC(C#C)(O)C2)=O)C2CCC2)cc(OC)c(F)cc1N C1(NC(C(C)C)=O)COC2(CNC(C3(P(C)(C)=O)CC3)=O)CC1C2 C1(CC)CCN(C(C2(F)CCCCC2)=O)C1CNC(=O)CC1CCCC(C)C1 CC1COc2c(NC(C3CCC4(C3)CC4C(=O)O)=O)cnn2C1 C(CC(C)C(=O)N1CCN(C(=O)CNC(=O)CN2CCCC(CO)C2)CC1)OC CC(C)(C)C(CO)C(=O)NCC(C)(C)NC(=O)CC1NC(=O)CNC1=O CCC(O)C(F)(F)C(=O)NCCC1(O)CN(C(=O)CN(C)C2CC2)C1 N1(C(CCC2(C)N=N2)=O)CC2(C(=O)NCCC3CCOCC3)CC1CO2 C1(N(C(CCC#C)=O)CC)CCCN(C(=O)CCn2cc(Br)c(C)n2)CC1 c1(OC)cc(CNC(=O)COC(C)(C)CNC(=O)Cn2nccn2)ncn1 CC(=O)C(C)CC(C)C(=O)N1CCC(C(=O)NC2(C(N)=O)CCC2)C1 c1(CNC(C(CN(C)C)NC(C)=O)=O)ccccc1-n1cc(C(C)(C)CO)nn1 C1(C(C)(C)C)(C(=O)NCC(CN(C(CCc2c(C)ncs2)=O)C)O)CCCCC1 C1(CC(=O)NC(C)(CO)C2CC2)C2CN(C(C3CC3(F)Cl)=O)CC12 c1(CC)c(C(=O)NCCNC(=O)C(CC2CC2)CC2CC2)nnn1CC C=C(Cl)C(C)(C)C(=O)N1CCC1CNC(=O)C(c1cccc(F)c1)(C)O C1(C(N(C(c2ccccc2)CC)Cc2cccnc2)=O)NCCC12CCOCC2 C1(O)(C(C)NC(c2cnn(CC(F)F)n2)=O)CCN(C(C2(F)CCOC2)=O)CC1 C1(CNC(C2(OC)CC2)=O)CN(C(C2CCCC2)=O)CCC1C n1(CC(=O)NC(CC=C)CNC(=O)C(CC)CC)nc(C(F)(F)F)c2c1CCC2 Cc1nc(N)c(CC(=O)NC2CCCCN(C(C3CN(C)C3)=O)C2)c(O)n1 C1(OC)(CNC(=O)C=CCC(C)(C)NC(=O)CCC2CCCC2)CCOC1 c1(C(=O)NC(CCNC(CN(C)CC)=O)C)sc(C2CC2)nc1C(F)(F)F C12(CNC(CCOCCOC)=O)CCCC1N(C(=O)CC1COCCOC1)CC2 N1(C(C(C(=O)OC)C)=O)CC(CNC(=O)COc2ccccc2)CC12CCC2 Cc1c(C(=O)NCCCN(C)C(c2cnn(C)c2Br)=O)cnn1CCN(C)C C1(CNC(C(C)(F)F)=O)CC2(CCN(C(=O)CSc3cccc(Cl)c3)C2)CO1 CCCCC(CC)C(=O)N(CC(C)(C)NC(c1nn(C)cc1Br)=O)C N1(C(=O)NC2CC(C)N(C)CC2)CCC2(CCCN(C)C2)C1 C1(C(=O)NCC(COCC)O)CCC(C)N(C(c2ccc(O)nc2)=O)C1 c1(OC)nc(C(=O)N(c2cccc(C)c2)CCNC(C)=O)sc1C Cc1cc(=NCC(C)(C)CCCO)[nH]c(=NCCCC2CC2(Cl)Cl)[nH]1 C1(NC(CCC=CCC=C)=O)CCCC(N(C)C(C2CCCCCC2)=O)C1 CCN(CCC#N)N1CCN2CCS(=O)(=O)CC2C1Cc1ccccc1 C1(C(=O)NC(C)COCC(F)(F)F)C2CCCC1N(C(c1sccc1C#N)=O)C2 c1(C(=O)NC(C2CCCN(C(c3cncs3)=O)C2)C)nc2n(c1Br)CCC2 c1(CC)ccc(C(=O)N(C2CCCN(C(=O)CC(C)COC)CC2)C)c(O)c1 C(=O)(C1=CC(C)(C)C1)NCC(C1CCN(C(Cc2ccc(C)nc2)=O)CC1)(C)O c1(CSCC)ccccc1C(=O)NC1CCCC1NC(=O)C(C)C1CCCC1 C1(C(N2CC(C(C)NC(C3CCCC3O)=O)C2)=O)CC12CC(C)(C)C2 C1(OCC)CN(C(c2cccc(Cl)c2)=O)CC1CNC(=O)COCC1CC1 C1(CC=C)(NC(=O)Cc2ccon2)CCN(C(=O)C(C)CC2CCCO2)C1 c1(Cn2c(-c3ccsn3)nc(C(CCC)C)n2)ccc(F)c(F)c1 n1(CC(=O)OCC(c2ncn(C)c2)=O)cc([N+](=O)[O-])cn1 C1(NC(=O)Cc2cn[nH]c2)CCC(NC(c2scnc2Br)=O)C1 CN1CCCC(C(=O)NCC2(C(N)=O)CN(C(=O)C(CC3CC3)CC3CC3)C2)C1 C1(C(=O)NC(CNC(CCN(C)CC)=O)(C)CO)CCc2nc[nH]c2C1 c1(CC(=O)NC2CCCC2NC(c2csc(Br)c2)=O)cnc(C2CC2)[nH]1 c1(C(N2CCC(N(C(C(CC)OCC)=O)CC)C2)=O)ccc(F)c(O)c1F Cc1cnc(C(=O)NCC2CC3CCC2N3C(c2n[nH]c(C)n2)=O)c(C)c1 c1(CCC(=O)NC2CC(NC(C3N(C(C)C)CCC3)=O)C2)nc2ccccc2[nH]1 c1(C(N(C(c2cccc(F)c2)C)CC)=O)cc(OCC)ccn1 C1(C)(C(C)C)CN(C(=O)C(C)OC2CN(C(=O)OC(C)(C)C)C2)CCO1 c1(OC)c(C(N2CCCC(CNC(=O)C(C)C3CC3)CC2)=O)ccc(Cl)c1C CCC(CC(=O)NCCCCCNC(C1C=CCC1)=O)C(=O)OC(C)(C)C C1(OC)CC2CC(C(c3nnnn3CCCF)NCc3nnc(O)o3)CC12 c1(C(N2CC(CO)C(O)C2)=O)n[nH]c2c1CN(C(c1ccc3c(c1)CCC3)=O)C2 CCCCC(C(=O)N(C(C)CN(C(=O)Cn1cc(C(F)(F)F)cn1)C)C)C(C)C CC1CN(C2CC2)C(=O)CC1.C(C)(C)CC1CC1 CCCC(C)(C)CC(=O)NC1COCC1NC(=O)C(C)(O)C(F)(F)F CC(C(C)(C)NC(=O)C=Cc1ccoc1)NC(C1CCCN1C(=O)C(F)(F)F)=O C1(NC(=O)NCCn2c(C)ccn2)CN(C(=O)C(C)(C)C)CCO1 C(CCCCC(=O)NC1(CNC(c2ccc(C(F)F)cn2)=O)CCC1)=CC O=C(CC1CCN1Cc1cnc(-c2ccccc2)s1)N=c1cnc(I)c(Cl)[nH]1 c1(NCc2c(C)nc(Br)s2)cc2c(cc1O)CCCC2 C1(C(N(C)CCN(C)C2CC2)=O)CCCCN(C(=O)CC2CCC(C)(C)C2)C1 c1(COC)nocc1C(=O)NCCC1(C(=O)N(CC(C)SC)C)CCC1 C(=O)(C(O)CC(N)=O)NCC(C(N1CCC(CCF)CC1)=O)N(C)C C(=O)(C1=CCC(C)CC1)N1CCC(NC(c2cc(C)nnc2)=O)C1 c1(-c2cn(C3C(SC)CCC3)nn2)cccc2[nH]ncc12.C12C=CCN(C1)C2=O C1(NC(c2n(CC)nnc2)=O)CCN(C(c2ccc(N(C)C)c(F)c2)=O)CC1F C(=O)(CC(C)CC(C)C)N1C(CNC(CCCc2c(C)ccs2)=O)C=CC1 C1(NC(COCc2cc(C)on2)=O)C2CC1N(C(C1CCCN1N=O)=O)C2 C12(CNC(C(C=C)c3ccccc3)=O)CC(CN1C(=O)CCCc1cnn[nH]1)C2 c1(O)ccc(C(=O)N(CC)CC2CCN2C(=O)C(CCC)SC)cc1.CCCCC=C c1(C(N2C(C)CC(NC(C3(C(=O)N(C)C)CC3)=O)C2)=O)cc(F)cc(Br)c1F C(CC(=O)NC1CC=C(C)CC1)(C(C)(C)C)NC(c1cnn(C(C)N)n1)=O CC1(C(=O)NCCOCCCNC(C2SCCS2)=O)CS(=O)(=O)C1 CCC(CC(=O)N(C)CC1(NC(c2ccn(-c3ccccc3Cl)n2)=O)CC1)SC CC(CC(=O)N1CC(F)(C(=O)NCC(O)(CO)CO)C1)C(F)(F)F c1(C(N2CC(C)N(C(=O)CC3(C)OCCO3)CC2)=O)ccn2nccc2n1 c1(CC(N2C(CNC(CC(C)SC)=O)CCCC2)=O)c[nH]c2c(C)cccc12 c1(C(=O)NC2CCCN(C(c3ncccn3)C)CC2)cc2ncccc2[nH]1 C=CCCN=C(NCC(=C1CCCC1)F)N1CCC(C(=O)OC)C(F)C1 C(CCC(C)(C)C(=O)N1CCN(C(c2[nH]nnc2C)=O)CC(C)C1)OC CC(C(=O)NC1(C(=O)NC2CC=CC2)CC1C)n1cncn1 c1(C(N2CC(CN(C(c3nc(C(C)C)oc3)=O)C)C2)=O)cnc(O)nc1O CC1(C(=O)NC2CCN(C(=O)CNC(=O)CN(C)C)C23CC3)CCS(=O)(=O)CC1 N1(C(CCC=C)=O)CC(NC(c2csc(Nc3ccccn3)n2)=O)C(C)C1 C(=O)(C(O)CCCNC(C1CCOCC1)=O)N1CC(C=C)C1 c1(C(=O)NCC(C(C)C)Nc2c([N+](=O)[O-])cnn2C)cc2c(s1)CCC(C)C2 C=CCC(C)(C)CNC(C1CCC(CNC(c2ccc(F)cc2)=O)CC1)=O Cn1nnc2cc(C(=O)NCC3CCN(C(=O)Cc4cnc[nH]4)C34CC4)sc12 C(C)(C)(CC(F)C(=O)N1CC2CCCC2C1)NC(c1cn(CC=C)nn1)=O N1(C(CN(C(=O)OCC)C)=O)CCC(NC(=O)C2CC2)CC1C.c1ccsc1Cl C1(C)(CN(C)C)CCN(C(c2coc(CO)c2)=O)CC1.C1(c2cscn2)C(=O)N1 C1(F)(CNC(c2cc(CCC)oc2C)=O)COCCN(C(C2(F)CCC2)=O)C1 N1(C(C(c2ccccc2)OC)=O)CCOCC1CNC(c1ccc(C2CC2)o1)=O c1(C(N(C(CNC(Cc2c(C)noc2C)=O)C)C)=O)cc(C(F)(F)F)ccc1N C1(NC(C2(S(N)(=O)=O)CC2)=O)CN(C(=O)C(C2CCCCC2)O)CCC1O N1(C(C(C(=O)OC)C)=O)CC2=C(C1)CN(C(=O)C1=COCC1)C2 CN1C(=O)CSC1=CC(=O)NCCC(O)CNC(=O)CCn1cccn1 CC1CN(C(c2ccc(Cl)s2)=O)CCC1N(C(=O)CCc1ccc(F)c(F)c1)C c1(-c2cc(OC)c(Cl)nc2)cc(C(=O)NCC23CCN(CC2)C3)c2cc[nH]c2c1 C1(C(N(CC(O)CO)C)=O)CCCN(C(=O)CCCN2CCCC2)C1 c1(C(=O)NC(C2(O)CN(C(c3cc(CC(C)C)on3)=O)C2)C)cc(Cl)cnc1O C1(C)(CNC(C2(COC)CCC2)=O)CN(C(=O)CCc2cnoc2)CCO1 C(=O)(C(O)C(F)(F)F)NCC(C1CCCCC1)NC(c1sc(CC)c(C)c1)=O Cc1ccc2c(=NC(C)C3CSC3)[nH]c(=NCC(=O)N3CCCO3)[nH]c2c1 Cc1cc(Cl)cc(C(N2CCC(NC(=O)CC(C)CN(C)C)CC2)=O)c1N N1(C(C2(C#C)CCC2)=O)CCCC(NC(c2cnc(CCC(F)(F)F)s2)=O)C1 c1(CCC2CN(C(=O)NCc3ccc[nH]3)C2)ccccc1 c1(C(=O)OCC)c(C)[nH]c(C)c1S(=O)(=O)NC(CCc1ccccc1)C(N)=O C1(NC(C(C)N(C(C)=O)C)=O)CCCC12CN(C(c1cccc[n+]1[O-])=O)C2 CC(C)(CNC(=O)C1=CCCSC1)CC(=O)NCC1(C)CC1(C)C C1(CNC(c2cn(C(C)(C)C)nn2)=O)CN(C(c2ccsn2)=O)CC1(C)C C1(CC=C)(NC(c2cnn(-c3cccc(Cl)c3)n2)=O)CCN(C(=O)CC2CC2)C1 C1(C(=O)NC(C2CC(NC(c3c(OC)n(C)nc3)=O)C2)C)CC1C1CCCC1 N1(CCSCC(=O)N(C2CC2)CC)CC2CC1CC2N1CCNCC1 CC(CC(=O)N1CCC(CCNC(=O)C(F)(F)C2CC2)CC1)CC(C)(C)C CCCCS(=O)(=O)CC(=O)N1CC(NC(=O)Cc2ccc(OCC)cn2)CC1C C(N=c1ccc(C(F)F)n[nH]1)C1CC(OC(C)(C)C)C1 C(=O)(CCCCC(F)(F)F)N(C1CCN(C(c2cc(C(N)=O)no2)=O)C1)C c1(C(=O)OC)cc(C)c(C(=O)NC2CN(C(C3CCOCC3)=O)CC2C)o1 c1(C(=O)NC2CN(C(C(C=CC)O)=O)C(C)(C)C2)oc2ccccc2c(=O)c1C c1(CC(=O)O)ccc2nc[nH]c2c1.C1(N(C)C)C2CN(C(=O)COCP(C)(C)=O)CC12 C(=O)(CCC1=CCCCC1)N1C(C(=O)NCC2CC(C#N)C2)COCC1 CC1CCN(C(=O)C(=O)NCc2ccc(=NCc3ccccc3)[nH]c2)CCS1 C1(CN(c2cc(NC(C)CC(N)=O)ncn2)C)COc2ccccc2O1 c1(C(=O)NCC(CNC(C2C(C)OCCC2)=O)O)cnn2ccccc12 c1(CC)cc(NC(N2CCCC(C)C2C)=O)c(C)nn1 C1(CCNC(CC(C)O)=O)CCCCN1C(c1ccccc1OC1CCCC1)=O c1(NC(c2nc(C(=O)NCC)sc2)=O)cc(NC(=O)OC)c(C)cc1Br CC(C)C(C)CC(=O)N1CCC(c2cn(-c3cccnc3C(=O)O)nn2)C1(C)C C1(C(N2CCC(COC)(NC(C34CC(F)(C3)C4)=O)C2)=O)COCC(=O)N1C(C)C c1(CC(=O)NC(CNC(c2c(C)ccs2)=O)(C)CO)ccc2c(c1)NC(=O)C2 N1(C(c2c(C)cno2)=O)CCC(C(F)(F)F)CC1CNC(=O)CCCC1CC1 C(=O)(CC1=CCCC1)Sc1c(CN2C(C)COCC2)cccc1 N1(C(C)C(=O)N2CCC2C(N2CCC(Cc3nccs3)C2)=O)CCOCC1=O c1(NC(c2ccsc2)=O)ccc2c(c1)CCN(C(=O)C1=CSCS1)C2 C=CCC(C)(C)CCNC(=O)C(n1cc(C2(C(C)C)CC2)nn1)C C(CC(F)F)(C(=O)NCCN1CCC(O)C1)N(C(=O)Cc1cc[nH]c1)C CC#CC1CCN(C(C2(CCNC(=O)C(C)NC(C)(C)CC)CCC2)=O)C1 c1(CC)ncccc1C(=O)N(C(C)C(=O)NC(CN(C)C)CC(C)C)CC C1(NC(C(C)C2(O)CCC2)=O)CC2CCCC(C1)N2C(c1ccc2c(c1)CC2)=O C(=O)(C(C)C(=O)N1CCC(C(=O)NCC(C)(C)CC2CC2)(CO)C1)OC C1(CNC(c2n[nH]c(C)c2C)=O)CCN(C(=O)Cc2cccs2)CC1C C1(C)(C(=O)OC)CN(C(=O)NCCc2c[nH]c3cnccc23)CC1(F)F c1(NC(NNC(C(C)(C)C)=O)=O)cc2c(cc1Cl)NC(=O)C2.c12ccccc1SCC2 Cc1cc(F)c(N)cc1C(N1CC(N(C)C(c2ccon2)=O)C(F)C1)=O c1(OCC)cccc(C(=O)NC(CNC(=O)COCC(F)(F)F)C(C)(C)C)c1 Cc1ccc(C(=O)NCC2(C)CCCN2Cc2ccccc2CO)cc1[N+](=O)[O-] C(=O)(CC1NC(=O)c2ccccc21)N1CC(c2cn(-c3ccc(CC)cc3)nn2)C1 C(=O)(C(O)CCSC)NCCN(C(CCC1N(C)CCC1)=O)Cc1ccccc1 c1(C(N2CCC(CNC(C3(O)CCC3)=O)C2)=O)cnc(O)c2ccccc12 c1(C(N(C(CCNC(Cn2cccc(C)c2=O)=O)C)C)=O)n[nH]c2cccnc12 C(=O)(CN=c1cc[nH]cc1)N1CCN(C(CC2C(C)C(=O)CC2)=O)CC12CC2 Cn1cc(NS(=O)(=O)C2CC2)cc1C(=O)Nc1n[nH]c(C(F)(F)F)n1 CCC(CNC(C1(C(F)F)CCCO1)=O)(CC)NC(c1coc(C(C)OC)n1)=O N1(C(=O)CCc2sccc2Br)CC2CC(NC(C3(CCO)CC3)=O)CC1C2 C(=O)(C(C)(C)C1CCOC1)NCCN(CC)CC1CCOCC1 Cc1cc(C(=O)NCCCC(C)NC(=O)Cc2ccc(O)cc2Cl)c(O)nn1 N1(C(C(CCC)CCC)=O)CC2CCN(C(=O)CC(C)OC)CC2C1 c1(C(=O)NC(C2(O)CCN(C(CC(=C=C)C)=O)C2)C)c(OC)cc(OC)cc1F c1(C(N2C(CC)C(C(=O)NC(C)CCC(C)C)CC2)=O)cc(O)ccc1C c1(C(C)NC(C(C2CCN(C(=O)CC3CC4(CCC4)C3)C2)C)=O)ccccc1F CC1CCN(C(=O)Cc2n[nH]cc2Br)CC1CNC(=O)Cn1cnnc1O c1(C(N2CCC(C(=O)OC)C2C)C(=O)NC(CC)C)cc(S(N)(=O)=O)cs1 C1(CC(N(C)C[Si](C)(C)C)=O)C2CCCC2N1C(=O)Cc1ccncc1 c1(CNc2ccc(-c3cc(OC)c(O)cc3Br)cn2)ccc(F)c(S(C)(=O)=O)c1 c1(C(=O)NCC2C3CN(C(c4cnc(C)s4)=O)CC32)cc(O)cc(=O)o1 C1(C(=O)NC(C2CN(C(c3csnc3Cl)=O)C2)C)CCC2CCCCC2C1 C(=O)(C(C(=O)NCC(O)CN(C(=O)C=Cc1c[nH]nc1C)C)OC)OC Cc1c(Br)c(CC(N2CCCC(C(N3CC4CC3CS4=O)=O)C2)=O)nn1C Cc1nc(Cl)[nH]c(=NCC(C2CC2)NC(C2CCC(F)(F)CC2)=O)c1F C(=O)(C(C)S(C)(=O)=O)NC(CCSC)C(=O)NCC1CCCN1C c1(C(=O)NC2(C(=O)NCCCCNC(N)=O)CC(F)C2)ccn2nccc2c1 C1(NC(C(CCC)O)=O)COCCN(Cc2ccc(C)cc2)C1 c1(-n2cc(-c3nc(C(=O)OC)c(C)s3)nn2)ccc(OC)c(F)c1 c1(C(=O)NCCC2(O)CCN(C(c3c[nH]ccc3=O)=O)C2)ccc2nn[nH]c2c1 O=C1c2ccccc2C(=O)N1CCC(O)CNCC1(CN2CCCCC2)CC1 C1(C(=O)NCc2nc(C)c(Br)s2)CC12CCN(C(=O)C(=O)C(C)C)C2 C(=O)(C(CC)(CC)C(=O)OC(C)(C)C)N1CC(CNC(C2CC(C)(CC)C2)=O)C1 N#Cc1ccc(C(N2CC3CCC(C2)N3C(C2OC3CCC2CC3)=O)=O)c(O)c1 c1(CO)ccc(CCOCCOCCNC(C2CC(NC(C)=O)C2)=O)cc1CO C1(NC(c2cc(C)ns2)=O)C2CCN(C(=O)CC3CCCNC(=O)C3)CCC12 c1(C(=O)OC(C)C(=O)Nc2cc(CCC)ncc2)cc(CC)cc(C)c1 C1(CN(C(CC(=O)OC)=O)C)CN(C(C2(c3cc[nH]n3)CCC2)=O)CC12CC2 C1(C(F)(F)F)(C(N2C(CNC(C3CC(C)(F)C3)=O)CCC2)=O)CC2(CCC2)C1 C12(C(=O)NC3CCC(C(=O)Nc4ccc(C)nc4)C3)CCCN(CC1)C2 c1(C(N2C3(C(N(CC(=O)OC)CC)=O)CC(C2)C3)=O)cccc(O)c1C C1(NC(c2c(C)scn2)=O)CC2CCC1CC2NC(=O)CC1CCCOC1 N1(C(CC(C)(C)SC)=O)CCC(C2CCCN(C(C3C=CCCC3)=O)C2)CC1 C(=O)(C(CC(=C)C)NC(C1(C2CC2)CC1)=O)Nc1cccc(CC=C)c1 CC1CN(C(C2(CO)CC2)=O)CC(CCNC(=O)CC(=O)Nc2nccs2)O1 N1(C(C2CCC(=C)CC2)=O)CCCC(CNC(=O)CC2CC3CC3C2)CC1 N1(CC(=O)N(CC)CC)CC2CCCN(C(=O)C(F)CC3CCCCC3)C2C1 CCCC(C(=O)OC)C(=O)NCC(C1CCCCC1)NC(=O)C1=C(Cl)CCCC1 CCCCCCCCCC(=O)N1CC(NC(C2CCCN(CC)C2)=O)C(C)C1 c1(C(=O)NC2CC(CNC(C(C)(C)OCC)=O)C2)nn(CC)cc1Br Cc1cn2cc(C(=O)N(C(CNC(=O)C(C)(C)CF)C3CC3)C)ccc2n1 Cc1cccc(-c2cn(CCN(C)C(c3cccnc3CC(C)C)=O)nn2)c1C C=C(C)CC(C(=O)NCCC1(C)CCN(C(=O)C(O)C(C)CC)C1)OC C1(NC(C2(OCC)CCCC2)=O)CCCC(NC(=O)CC(C)N2CCCC2=O)C1 N1(C(CCSCCCC)=O)CC(CNC(=O)CS(=O)(=O)CCC)CC(C)(C)C1 N1(C(C(C)n2ccnc2)=O)CCC(C)C(CC(=O)N(CC(C)(F)F)C)C1 CC(C)CCCCCC(=O)N1C2CCC1(CNC(C1(CO)CCCCC1)=O)CC2 C1(CNC(C2(C(=O)OC)C(=C)CC2)=O)CCCN(C(=O)C(CC)n2ccnc2)C1 c1(OC)ccc(Cl)cc1CC(=O)NC12CCN(C(=O)Cc3nnc(C)s3)CC1C2 CN1CCC(C)(C(N2CCC(N(C(=O)C3=NOC(C(C)(C)C)C3)C)CC2)=O)C1=O c1(SC)c(C(N2CCCCC2c2n[nH]cc2N)=O)cccc1[N+](=O)[O-] c1(C(C)(C)NC(c2ccc(C(=O)OC)cc2)C(C)C)ccc(F)c(F)c1F Cc1nsc2ncc(C(=O)NCCC(O)CNC(=O)CSC3CC3)cc12 c1(C(=O)NC2CN(C(C(C)NC(COC)=O)=O)C(C)(C)C2)ccc(Cl)c(C)c1N C1(CCC)CN(C(=O)C=Cc2ccccc2Cl)CCN1C(=O)C(C)OC(C)(C)C N1(C(Cc2cc(C)ns2)=O)CCC(C)N(C(=O)C(C)C(F)(F)F)CC1 C1(C(C)NC(C2(C=C)CC2)=O)CN(C(c2cnn(CCC)c2)=O)CCO1 N1(C(C2(C#C)CCCC2)=O)CC2(CC(NC(=O)C3=CC(C)(CC)C3)C2)C1 c1(CC)c(C(=O)N(CC(C)CNC(C2(F)CCOC2)=O)C)sc2ccccc12 c1(C(=O)NCCNC(c2c(CC)noc2C)=O)ccc(C(F)(F)F)c(O)n1 C1(C(N(CC(C)(C)CNC(C2C(F)(F)C23CC3)=O)CC)=O)CC(C)(C)OC1(C)C CCCCC(C)C(=O)NC(CO)C(C)NC(c1ccc(C(N)=O)[nH]1)=O c1(C(=O)NCCC2C(C)CN(C(=O)Cc3ccsn3)C2)ccc2[nH]ccc2n1 C1(C(=O)NCCCOC)COCCC12CCN(C(=O)Cc1ccccc1C)CC2 c1(C(C)=O)cncc(C(N2CCC(O)C2C(N2CC3CC2CO3)=O)=O)c1 N1(C(C2CC(OC)C2)=O)CCOCC1CCNC(c1cn(C2CCOC2)nn1)=O c1(NC2C(CF)CCC2)nc2c(c(=NC3CC4CCCC4C3)[nH]1)CSC2 C1(N(C(COC(C)C)=O)C)CCCC(NC(C2CCCN2C)=O)C1 N1(C(CNS(CCCC)(=O)=O)=O)CC2(C1)CN(C(c1cncc(C)n1)=O)CCO2 CC(CC(=O)NCC1CCN1Cc1cc(C2CC2)no1)C1CCOC1 C(=O)(C#CC1CCOC1)NCC(C(C)(C)C)NC(c1c(NC)nc(C)cc1)=O C12(C(N(CC(CN(C(C3(C#C)CCCC3)=O)C)O)C)=O)CCCN(CCC1)C2 c1(C(=O)NC2C(NC(c3ccc(OC)cc3F)=O)C2)cnn2c1NCCC2 c1(NC(CC=C)C)cc(N2CCC(c3nncn3C(C)C)CC2)nc(C)n1 CC1CCN(CC(=O)N(C2CCCC(NC(c3cnc(C4CC4)s3)=O)C2)C)CC1 N1(C(c2n(C(C)C)ccc2)=O)CC(NC(c2nnc(C(F)(F)F)s2)=O)C(C)(C)C1 CC1CCCC1(C(=O)NCCOc1ccccc1)NC(=O)Cc1cccnc1 c1(NC(c2cccnn2)=O)cnc2c(c1)CN(Cc1cccc(F)c1I)CC2 C1(NC(=O)C=C2CCCCC2)CCC(O)CN(C(=O)CC2CCS(=O)(=O)C2)C1 C1(C(=O)NCCC(C)NC(c2csc(NC(=O)C(C)(C)C)n2)=O)C(Cl)(Cl)C12CC2 N1(C(C2CCN(C)CC2)=O)CCOC2(CCN(C(=O)CC34CC(C3)C4)CC2)C1 Cc1c(C(=O)NCCNC(=O)C(C)CC(C)C)ccc(Br)c1Cl C(=O)(CC(F)(F)CC(=O)NC1CCCCC1NC(c1c(C)nsc1C)=O)OC C1(F)(C(=O)NCC(C)NC(CCCCc2ccc(C)cc2)=O)CCCN(C)C1 C1(C(=O)OC)C(NC(c2nnnn2CCN2CCCC2)C2CC2)C2CCCCC12 c1(C(=O)NCCC(CNC(C(CCOC)C)=O)O)ccc2nnn(O)c2c1 c1(OC)coc(CSc2nnc(SC(C)C)n2-c2cccc(O)c2)cc1=O CC1CCN(C(=O)CC2CCCN2C(C2CC(C)(C)CO2)=O)CC1(F)F C(=O)(CCCCCOC)NCC(=O)OC1CN(C(=O)NCCOC)C1 C(=O)(CCCC(N)=O)NCCC1(C)CCN(C(c2cnc(-c3ccsc3)s2)=O)C1 c1(C(=O)NCCCN(C(C2(C)CCN(C)C2)=O)CC)cc(C)cc(C)c1 C1(c2n(C)ncc2)OCCCC1C(=O)NC1CC(NC(c2cn(CCF)nn2)=O)C1 C=C(C)CCC(=O)N(C)CCOCCCNC(=O)CC1(C(F)(F)F)CC1 N1(C(C2C(CC)CN(C(c3cnn(C(C)C)c3)=O)C2)=O)CCN(CC)C(=O)C1 c1(C(=O)NC(CNC(c2cc(C(C)C)[nH]n2)=O)C2CCC2)cc2cccnc2s1 n1(CC)nncc1C(=O)NC1(CO)CN(C(C2CC2c2sccc2C)=O)C1 N1(C(COc2cc(C)on2)=O)CCC2(CCC2)C(CNC(=O)C2=COCCC2)C1 C12(CNC(c3cc(C(C)C)n(C)n3)=O)CC(CO1)N(c1nnc(C(F)F)s1)C2 CC1CN(C)CC(C(N2CCC2(C)CC(=O)NCC2(O)CCC2)=O)O1 C(CC(F)F)(C(=O)NOCCCC1CC1)N(C(c1cc(OC)ns1)=O)C c1(C(=O)NC(CC(C)NC(c2nc(O)[nH]c(=O)n2)=O)C)cnc2c(c1)CCCO2 C(=O)(C(CNC(=O)CCc1cnn(C)c1)C(C)(C)C)NCCNC(=O)OCC N1(C(c2c(COCCC(C)C)cccn2)=O)CCCC(C)(C(F)F)C1 c1(C(=O)NC2C(CNC(C3N(C)CCC3)=O)CCCC2)cnc2ncnn2c1O N1(C(c2c[nH]c3ccc(Br)cc23)=O)CCOC2CCN(C(C34CC(C3)C4)=O)CC12 c1(OC)c(CN(C)Cc2nnn(C(C)(C)C)n2)cccc1Br c1(N2CCC(c3ccc(=N)[nH]c3)CC2)ccnc2c(Br)csc12 N1(C(C2CCC(COC)C2)=O)CCC2(CCC(NC(=O)C3=C(Cl)CCC3)CC2)C1 c1(NC(=O)Nc2csc(Br)c2)nc2c(s1)CCc1ccccc1-2 C1(CC)CC(C)CCC1NCC1CCCCNC1 c1(C(N2CC(CNC(COC)=O)C(C(F)(F)F)C2)=O)cc(Cl)cc(C)c1OC C12CC3(COC1C3)N2C(c1c(C)coc1C(C)C)=O.N1(C(=O)C(C)O)CCSCC1 C1(CC)CC(C(=O)NCCc2ccns2)CCN1C(=O)C(C)N(C)C(C)=O C(=O)(C(Cc1ccoc1)NC(=O)CCc1ncnn1C)N(CCN(C)C)C c1(NC(c2c(NCc3c(N)cccc3F)c[nH]n2)=O)cc2c[nH]nc2cc1F CCC(C)CC(C(=O)N(CC(C)SC)C)NC(c1cnncc1OC)=O N1(C(C(C)S(C)(=O)=O)=O)CC(C2CCCN(C(=O)CN3C(=O)CCC3=O)C2)C1 C(=O)(C1=CCCCO1)NCC(N(C)C(C1(C(F)F)CC1(F)F)=O)C1CC1 c1(CCC(=O)NC(CNC(=O)CCNC(c2ccco2)=O)C2CC2)cc(Cl)no1 c1(OCC(=O)NCCCCCNC(C2(C(C)C)CCC2)=O)ccc(F)cn1 C(CC(C)(C)C)(C(=O)N1CCC2CCCC12C(N1CCC(OC)C1C)=O)OC c1(-c2n(C(c3ccncc3)C)ccn2)ccncc1-c1cccc(F)c1 C(C(C)(C)C(=O)NCC1CC(NC(=O)Cc2cn[nH]c2)CC1O)N(C)C C1(CC)CN(C(c2occ(C)c2C)=O)CCN1C(c1ncc(C)cc1Br)=O CC1(C)CCCC(O)(C(=O)NCC2(NC(=O)CC3(CO)CC3)CCCCC2)CC1 c1(CC)cccc(C(N2CCCC2CCNC(c2cccnc2OC)=O)=O)c1N C1(C)(C(N2CCC(SC)C2)=O)CCN(C(=O)C(=O)NC2CC2)CC1 CC1CN(C(=O)Cn2cnnn2)CC1CNC(=O)C(C)(C)C1(O)CCOC1 Cc1cc2n[nH]cc2cc1C(=O)NCCCCCNC(=O)Cn1ncccc1=O CC#CCCC(=O)NCC1COCC1NC(c1cc(CC)nn1C)=O C12(CNC(=O)Cc3ccc(Cl)nc3)CCCC1N(C(c1cc(=O)cco1)=O)CC2 n1(COCC)nnc(C(N2CC(CNC(=O)C=C(C)C(C)(C)C)C3CC23)=O)c1N CC(CCCNC(=O)C(C)NC(N)=O)NC(=O)CC1CC(=O)C1 C1(NC(Cc2c(C)nc[nH]2)=O)CCCC12CCN(C(C1(C)CC(F)(F)C1)=O)C2 C1(C(=O)NC(C(N2CC(C#N)C2)=O)CC2CC2)CC(N=[N+]=[N-])C1 C1(OC)CC2(C1)CC(C(=O)OC(Cc1ccccc1)Cc1ccccc1)C2 N1(C(c2cc(CC)[nH]n2)=O)CCCC(CCCC(=O)NCC2(C)CCCCO2)C1 c1(COC)c(C(N2CCN(C(C3(Br)CC3)=O)CC23CCC3)=O)oc2ccccc12 C1(CC)(CC)CC(NC(=O)CSC(F)F)CN1C(C1C2CCCOC12)=O c1(CC=C)cccc(C(=O)NC(C)C(C)NC(=O)CCC2CC(OC)C2)c1 c1(C(=O)NCCCCN(C)C(C2CCCOCC2)=O)cc(F)cc2c1CCC2 Cc1nc(NC(c2cc(C(C)(C)C)on2)=O)c(F)c(Cl)n1 N1(C(c2c(CC)ccs2)=O)CC2(CNC(=O)C(C)Cc3ccco3)CC(F)(C1)C2 N1(C(Cc2c(C)n(C)nc2)=O)CCN(C(c2ccoc2C2CC2)=O)C(CCO)C1 C(=O)(CC(C(C)OC)NC(C1CC(=C2CC2)C1)=O)NC(CCC)C1CCC1 N1(C(CP(C)(C)=O)=O)CC(NC(c2occc2Br)=O)CC2(CC2)C1 CC(C)CC(C(=O)NOC(C)(C)C)ONC(=O)C1(CCF)CCC1 C1(NC(c2ccc(C)cc2Br)c2n(CCSC)nnn2)CCCC(C)(C)C1 CC(=NO)C1CC(C(=O)NCC2CN(C(=O)C(O)CCc3ccccc3)C2)C1(C)C C=CCC(CNC(C1CCOC1C(C)C)=O)C(=O)NCc1nc[nH]n1 c1(C(C(=O)NCC2C(NC(CSCC=C)=O)C2)=O)ccc(Cl)cc1 c1(C(C)(C)C)ccc(OCCNC(C2CCC(=C3CCC3)CC2)=O)cc1Cl C1(C(=O)NCCNS(NC)(=O)=O)CC2(CCN1C(C1CCN(C)C(=O)C1)=O)CC2 C1(CNC(c2c(C)onc2)=O)CC2(CCN(C(C3CC3C(F)F)=O)CC2)CO1 N1(C(=O)OCC(C)C)CCC12CCC(F)(F)CC2 N1(C(CC2CC(=O)NC2)=O)CCC(O)(CNC(c2nocc2C(C)(C)C)=O)CC1 C1(CC=C)(C(=O)NCCC(C)CC)CCCN1C(c1cc(C(F)F)[nH]n1)=O N1(C(c2nc(CC)oc2C)=O)CCC2(CC2)CC1C(N1CC(C(=O)N(C)C)C1)=O c1(SC)cc(F)ccc1C(=O)N(CCCN(C(=O)CC1(N2CCCC2)CC1)C)C C1(NC(C2CCC(C)CC2)=O)CS(=O)(=O)C12CCN(C(C13COC(C1)C3)=O)CC2 C=Cc1ccc(C(=O)NCC2C(C)CCCN2C(=O)C(C)OCC)cc1 C1(N(C(C2C(=C)CC2)=O)CC)CCCN(C(C2(c3cncnc3)CCCC2)=O)CC1 c1(CC(N2CC(O)(CNC(C3C(C(=O)OC)C3)=O)C2)=O)cccc(C)c1 N1(Cc2ccc(SC)[nH]2)CCCCC12CCCCC2 C1(NC(C(CC)(C)CC)=O)CC2CCC(C1C)N2C(=O)CCCn1cccn1 CCC(O)CC(=O)NCc1nc(C)c(C(=O)NCCC2(C)N=N2)o1 CCCCCC(O)C(=O)NCC1CN(C(c2c[nH]c3ccccc23)=O)CC1C c1(C(=O)NCCCCCNC(=O)COC2CCC2)cnc2cccnc2c1 C12(C(=O)NCCC(COC)OC)CC(C)(CN1C(C1CCC(N(C)C)C1)=O)C2 c1(OC)cccc(C2CC2C(N2CCC(NC(=O)CC(C)OC)C2C)=O)c1 c1(NC(CC2(NC(C3CC(CCC)C3)=O)CCC2)=O)cn(C)nc1O N#Cc1ccccc1C(=O)NCCC1CCCCN1C(=O)CC(F)(F)F c1(C(=O)NCC2CCC(NC(c3n[nH]cc3F)=O)C2)cccc(Cl)c1F O=C(C#CC1(C(F)(F)F)CC1)NCC1CN(C(C2(F)CC2)=O)CCC1C(F)(F)F C1(NC(CC2CC(C)(C)C2)=O)CC(N=c2ccc(C(F)(F)F)n[nH]2)C1(C)C N1(C(C(C(CC)C)C)=O)CCN(C(c2ccncc2SCC)=O)CC(C)(C)C1 C1(NC(C2(CC)CCC2)=O)CC12CC(NC(=O)C(O)Cc1cnc[nH]1)C2 c1(OC)c(C(=O)NC(C)(CNC(c2csc(Cl)n2)=O)C2CCC2)occc1=O n1(CC)cccc(NC(=O)C(n2ccc(C)n2)C)c1=O C1(CC(=O)NC)(NC(CN(CC)Cc2c(CC3CC3)c(C)[nH]n2)=O)CCOCC1 N1(C(C2C(CC)OCC2)=O)CCCC1(CO)CNC(=O)CCc1cn[nH]c1 C=C(C)CCCC(=O)NC1(C)CCCN(C(c2nc(OC)ccc2OC)=O)C1 C(=O)(CC(C(F)F)C(C)(C)C)Nc1cc(C)c(NC(C2CCC23CCC3)=O)cc1 C1(CC(=O)N(C2C(C)OCC2)CCO)COCCN1C(C1CCC(N(C)C)C1)=O c1(C(=O)NCCN(C(=O)C(C)CC(C)C)CCC)cnc2[nH]ccnc1-2 C(C(C)C)(C(O)C(=O)NC1CCC(CCNC(=O)CN2C(=O)CCC2=O)C1)OC N1(C(C(C2CC(F)(F)C2)OCC)=O)CC(NC(c2csnn2)=O)C(CC2CC2)C1 Cc1cc(C)c2c(c1)N(C(=O)NCCOc1cccc(Cl)c1C)CCO2 C12CN(CC13CC3)C2=O.C1(c2cccs2)(NC(C(CC)SC)=O)CCOCC1 C(=O)(C1CCCc2n[nH]cc21)N1CC(O)(CCNC(c2ccc(C#C)cc2)=O)C1 N1(C(C(=O)NC(C)C)=O)C(C(=O)NC(C)C(=O)OC(C)(C)C)C2CC(O)C1C2 Cc1ccc(C(=O)CCC(=O)NCC(CO)NC(=O)C=Cc2ccccn2)cc1 CC1=NNC(=O)C1CC(N1CCC(OCCNC(c2nnc(S)n2C)=O)C1)=O c1(NC(C2N(c3nc(OC)c(F)cn3)CC(F)C2)=O)cc(Cl)cc([N+](=O)[O-])c1C Cc1cccc(C)c1NC(=O)C(CC(C)C)ONC(C1CCC2(CCC2)C1)=O C(N=c1[nH]cnc2cccnc12)C1CCC(CN(C(C(C=C)(C)O)=O)CC)CC1 C1(C(N(CCCC(C)C)C)=O)CCCCCC1NC(C1CCC1C(C)(C)C)=O C1(CC(=O)NCC2N(C(C(C)OCCC(C)C)=O)CC2)CCN(C(C)C)CC1 c1(N2CCC(NC(=O)NC3C4(CC(OCC)C4)C3)C2)cccc(F)c1F C(=O)(C1=CCCN(C(c2ccc3nc[nH]c3c2)=O)C1)NC(C(C)C)CO CN1CCC(CC(=O)NCCCC2(NC(C3CCN(CCF)CC3)=O)CC2)C1=O Cc1nc2ccccc2n1CC(=O)NC1CC1NC(c1c(F)ccc(F)c1F)=O c1(CC(N2CC(F)CC2C)C(=O)NCCCSCC)cc(Cl)c(Cl)s1 N1(CC)CCN(C(=O)Cc2cc(C)no2)CC1.C(CN(C(C)=O)C)OCC Cc1ccccc1C(N(C)CCN1CCN(C(C2CS(=O)C2)=O)CC1)=O S(=O)(=O)(c1ccc(C(=O)NC2CCN(C(c3ccc(C(C)F)cc3)=O)C2)o1)NC CCC(C)(C)CC(=O)NCc1cc(C(=O)NC(c2ccccc2)C)n[nH]1 C1(CC)(Cn2cc(CC(=O)NC3(C)CCCC3N(C)C(C)=O)nn2)CC12CCC2 c1(C(=O)NC(C(C)C)CNC(c2cncc(CO)c2)=O)cc2cccnn2c1 C1(CCC(=O)OC)CC(C)(C)CN1C(=O)C(c1ccccc1)F.c12nc(no1)C2 c1(NC(c2cc(CNC(C(C)SCCCC)=O)nn2C)=O)ccc(Cl)c(O)c1 C(=O)(CS(=O)(=O)CC)NC(COCC)C(=O)NC1(C2CCCO2)CC1 C(=O)(C(C)C(F)(F)F)N1CCC(C(C)NC(CCC=CC(C)C)=O)CC1 c1(OC)cc(C)c(C(N2CC3(CCC(CNC(C4CC4C)=O)O3)C2)=O)c(F)c1 C1(NC(c2cn(CC)nc2)C(F)(F)F)COCC1(C)C C1(CNC(c2ccc(CO)nc2)=O)CCCCN(C(c2ccccn2)=O)CC1 C(=O)(C(C)C(C)C(C)(C)C)NC(C)CCCNC(=O)C=CC(=O)N(C)C Cc1cc(=NCCCC(C)NC(C2CCOC3(CCCC3)C2)=O)[nH]c(C(C)C)n1 C1(NC(c2cc(COC)no2)=O)(CO)CCCN(C(C2(C)CC=CCC2)=O)C1 N1(C(N(CC)Cc2cc3ccccc3[nH]2)=O)CCc2nc(C)nc(O)c2C1 C1(CNC(C(C)(C)CC(F)F)=O)CCC2CN(C(c3cnc[nH]3)=O)CCC2C1 C1(C(=O)NCC2N(C(CN(CCC)C)=O)CCOC2)Cc2cccc(F)c2O1 Cc1cccc2nc(N3CCOC(C)(CNC(c4cocn4)=O)C3)oc12 C1(NC(C(CCCC)C)=O)CCCCCN(C(c2ncnc3ccsc23)=O)C1 Cc1ccc(C(C)CC(=O)NCCNC(C2CCCN(CC(F)(F)F)C2)=O)cc1 CCCCCC(CC)C(=O)NC(CNC(=O)C(F)(F)CO)CCOC C1(NC(Cc2c(OC)nccc2)=O)CN(C(c2nnccc2C)=O)CCC1F N1(c2c(C)ccc(Cl)c2)CCN(N2CCCC(C)(C)C2CO)CC1 c1(CN(C(C(=O)NC(C)C)C2CC2(C)Br)C2CC2)cccc(C(F)(F)F)c1 Cc1nsc(C(=O)NC2CC23CC(NC(C2CC(=O)N(C)C2)=O)C3)c1N C1(C)(NC(CC2CC(NC(CN(CCC#C)C)=O)C2)=O)CC(O)C1 c1(NC(CCOCCC)=O)cccc(NC(=O)CCC2C(=O)ON=C2C)c1 N1(C(c2nc(COC)oc2)=O)CC2(NC(=O)Cc3ccc(F)cc3)CCC1CC2 c1(C(=O)NC(C2CCN(c3ccnc(CO)n3)C2)C)cc2n(n1)CC(F)C2 c1(CCC(=O)NC2C(NC(C(C)c3cncs3)=O)COC2)cnc2ncccn12 N1(C(CCCNC(C)=O)=O)CCC(C)C(CC(=O)NCc2ccn(C3CC3)n2)C1 C1(C)(C(N(CCNC(Cn2c(C)ncc2)=O)C)=O)C2Cc3ccccc3C12 c1(-n2cc(C(=O)NC3C(CNC(c4cocn4)=O)C3)nc2)ccc(Cl)c(Cl)c1 C1(NC(c2c(C)nsc2)=O)CN(C(=O)Cn2cc(CO)nn2)CC1(C)C Cc1cc(CC(=O)NCCCN(C(C)C(=O)NC2CCOCC2)C(C)C)n(C)n1 c1(NC(c2n(CCC)nnn2)c2conc2C2CC2)ccc2c(c1)C(O)CC2 c1(C(=O)NC2C(NC(CCc3cc(OC)no3)=O)CC2)ccc2c(n1)CCOC2 CC1CC(NC(=O)C(F)C(F)(F)F)CCN1C(=O)C(c1ccc(C(F)F)cc1)=O c1(C(N2CCNC(c3ccc(Cl)cc3)C2)=O)c(O)cccc1Br N1(C(=O)COCC(F)(F)F)CCC2C(CCCN2C(=O)CCC2CCCOC2)C1 c1(OC)c(C(C)CC(=O)N(Cc2cn(C(C)C)nn2)CC2CC2)cccc1F C1(n2cccn2)(C(=O)NC(CC)CO)CCN(C(c2cc(O)n(C)n2)=O)CC1 Cc1nc(NC2CC2C2CC2C)cc(N2CCC(C)(OCCO)CC2)n1 N1(C(c2cc(CCC(=O)O)sc2)=O)CCCC(C(=O)C2CC2)C1 N1(C(C(O[Si](C)(C)C(C)(C)C)C)=O)CCC2(C1)CN(c1ccncc1)C2 C(=O)(CCC(=O)N1CCC(CC(C)NC(=O)Cc2cnccc2Cl)CC1)OCC C(=O)(C(C)Cc1cnn(C)c1)NCCCN(C(C(C)SCC)=O)C c1(C(=O)NC2CCOCC2NC(C2(CO)CCCC2)=O)cncc(OC(F)F)c1 C(=O)(CCCCC1CC1)N1CCC(CC(=O)NCc2[nH]nc(OC)c2Cl)C1 C1(C(=O)OC(C)(C)C)CC(NCC(=O)Cc2ccccc2F)C12CCOCC2 C1(NC(C2(NC(C(C(CC)O)C)=O)CCCCC2)=O)CC2(CCCC2)CO1 C12(C(=O)NCC3CN(C(=O)CCc4ccoc4)C4C3C4)CC3CCC(CC(C3)C1)C2 C1(OC)CCCCC1C(=O)NCCCC(C)(C)NC(=O)C#CC1CC1 CCC(CC(=O)NCC1CC(C)CN(C(c2cc(C(N)=O)cn2C)=O)C1)C(C)C C1(O)(c2cn(CCCCC)nn2)CCN(C(C2(c3cccs3)CC2)=O)CC1 C(=O)(CC1=CCN(C)CC1)NC1(CCCCNC(C(C(C)C)F)=O)CC1 CC(C)CC(C)C(=O)NC1CCCCC1NC(=O)C(c1cc(Cl)cc(Cl)c1)(C)C c1(NC(C=CC=CC)=O)cnn(C2CN(C(C3CC(O)C3)=O)C2)c1 CC(C)C(CC(=O)NCCNC(c1cc(CO)n(C)n1)=O)c1ccccc1 c1(CN2C3C(C(=O)Nc4ccc(C)c(Br)c4C)C(C3)C2)cc2cc(Cl)ccc2[nH]1 C(=O)(C1=NN2CCCN=C2N1)N1CCC(C)C(NC(c2cnsn2)=O)C1 c1(C(=O)NC(CN(C)C(c2cnn3ccccc23)=O)(C)C)ccc2cc[nH]c2n1 c1(C(=O)NC2C(CNC(c3c(C)sc(Cl)n3)=O)C2)cc([N+](=O)[O-])cn1C c1(C(C)NCc2ccc(-c3cccnc3F)cc2)ccc(O)c(Cl)c1 c1(NC(c2ocnc2C(F)(F)F)=O)cnc(C2CC2)cn1 N1(C(C(c2cncnc2)C)=O)C2CCC1CN(C(C1COC3(CCC3)CO1)=O)C2 CN1CC=C(CC(=O)NCCCCCCNC(c2ccc3nncn3c2)=O)CC1 N1(C(Cn2c(C)ccn2)=O)CCN(C)CC1CNC(c1cnc(O)c(F)c1)=O n1(CCN(C(C2CCN(CCC)CC2)=O)C(C)C)cnc2c(N)ncnc12 C1(NC(C2C(C)CCO2)=O)CC2CCC(C1)N2C(=O)C(C1CCC1)C1CCC1 c1(C(N2C(C)CC(CNC(=O)C(C)(C)c3ncco3)C2)=O)[nH]nc2ncccc12 CCCCCCCCCCC(=O)N1CCCCC(NC(=O)C(C)(C)OC(C)=O)C1 C1(NC(C2C(CCOC)C2)=O)CN(C(c2cnc(C)cc2C)=O)CCC1CO CCC(O)C(O)C(=O)Nc1ccc(OCC(F)(F)F)nc1 N#CC12CN(C(=O)C(CC3CC3)CC3CC3)CC1CS(=O)(=O)C2.c1nncs1 CC(C)C(C)C(CNC(=O)CC(C)(C)O)NC(c1cnc(C2CCOCC2)s1)=O C1(NC(c2cc(C)n(C3CC3)c2C)=O)CS(=O)(=O)CC1N=c1[nH]nc(C)s1 N1(C(C2CC(C(=O)OC)C2)=O)CCCC(NC(C2(C)CC2(C)C)=O)CC1 C12(CNC(C3CC(C(F)F)C3)=O)CCCC(CN(C(=O)C(O)C(F)(F)F)C1)C2 C1(C(N(CC(O)CO)C)=O)CC1C1CN(C(C2CC2Cl)=O)C1 c1(OCC=C)cccnc1C(N1CC(C)(NC(=O)CNCc2ccccc2)C1)=O C1(F)(C(N2CCC(OCCNC(c3cccc(C(F)(F)F)n3)=O)C2)=O)CC=CCC1 C(=O)(C(CC#CC)NC(=O)CCCCC#N)NC(C1CCCC1)C#C N1(C(C2C(C(N)=O)C2)=O)CC(O)CC1CC(=O)NCC1CN(C(=O)N(C)C)C1 C(C1OCCc2ccccc21)NCC1CCC2C(F)(F)C2C1 N1(CC2(NC(C=C(C)Cl)=O)CC2)CCN(C(c2[nH]cnc2C)=O)CC1 c1(N2CCCC(C)(COC)C2)ccc(S(=O)(=O)N(C2CCCC2)CCC#N)cn1 Cc1nc(C=CC(N2CC=CC2CNC(c2sccc2Cl)=O)=O)[nH]c1C C(=O)(C1=CC(C)(C)C1)NC1C(NC(c2nc(C)c(C)s2)=O)C1 CC1=NNC(=O)C1CC(=O)NCCN(C(C1CC12CC(O)C2)=O)CC1CC1 Cc1cc(C(N2CC(C(N3CCOC(C)(C4CC4)C3)=O)(C(C)C)C2)=O)cc(O)c1 S(=O)(=O)(c1ccc(NCCSC(F)(F)F)c(F)c1)NC1(C)CCC(C)C1 C(=O)(C(C)CC(=O)NC(C(=O)NCc1cnc(C)s1)C(C)(C)C)OC N1(C(C=CCN(C)CC)=O)CCCC(CN(C)C(c2scnc2C)=O)C1 c1(CC(=O)NC(CC)CNC(=O)C(c2cccs2)SC)csc(C(C)(C)C)n1 C=CCC(C(=O)NC(CCNC(=O)CCCOC)(CC)CC)C(C)C CC(C)CCC(=O)NCC1(O)CC(CNC(=O)CC2(O)CCCC2)C1 N1(C(C(C)N(C)C)=O)CCC(CNC(=O)CCC(=O)N(C)C)CC1C N1(C(C2CC(=O)C2)=O)CCC2(CCC(CNC(C34CCCC3C4)=O)OC2)CC1 O=C(C#Cc1ccc(C(F)(F)F)cc1)NC1CCCC(F)(F)C1 c1(CCC(N2CCC(CN(C)C(c3c[nH]nc3C3CC3)=O)C2)=O)nnc(S)n1C c1(C(N(C2C(NC(CSc3nc(C)[nH]n3)=O)CCCC2)C)=O)c[nH]c(=N)nc1C C(=O)(C1=CCCCO1)N1CCC(N(C(=O)CC2CCC3CC23)CCOC)CC1 C=CCCCC(C(=O)NCC(C)CCCO)NC(c1coc(OCC)n1)=O C(CC1CC1)(CC(=O)NC1CCS(=O)(=O)C1)NC(C1C(=C)C1C(=O)OC)=O C(=O)(CC(C)C(C)(C)C)N(CC(C(=O)N1C(C)(COC)CC1)(C)C)C C(=O)(C(C)CC(F)(F)F)N(CCCCCC)CCNC(C(CC#C)O)=O C1(C(N2CCC(N(CCC)C(C3CNC(=O)N3C)=O)CC2)=O)COC2(CCC2)C1 n1(CC(=O)NCCCOCCC=C)cc(CNC(=O)C(C)NC(N)=O)nn1 N1(C(CCSC)=O)CC(N=c2[nH]c(Cl)ncc2F)C(C)(C)C1 N1(C(CCOC)=O)CC2CCN(C(=O)Cn3nc(C)c(C)c3C)CC12 C(=O)(C1=C(Cl)CCCC1)N1C(CNC(C(C)n2cccn2)=O)C(C)(C)CC1 c1(OCC)cc(F)ccc1CNC1(c2nnnn2C)CCC(N2CCOCC2)CC1 CC1=C(C)CC(C(=O)NCc2ccc(C(=O)NC(C)C3CC3)s2)CC1 N1(C(C(COC)NC(C2CCSC2)=O)=O)CCC=CC1CO N1(C(=O)Nc2cc(C(c3cccc(F)n3)OC)on2)CCCC(N2CCCC2)C1 C1(NC(C(CC)F)=O)CCC12CCN(C(c1cccc(C3COC3)c1)=O)CC2 C1(CNC(C(C(CC)C)O)=O)CN(C(c2cncc(F)c2C)=O)CCC1(C)C c1(C(C(C)NC(=O)Cc2csc(C(C)=O)c2)NC(C=CC)=O)ccccc1OC C1(CNC(C2(CCC)CCC2)=O)CCC2(CN(C(c3ccc(N)c(N)n3)=O)C2)O1 N1(C(c2c(CC)cccc2)=O)CC2CC(NC(=O)Nc3ccccn3)CC2C1 C1(NC(C2(C)CCC(=O)CC2)=O)CC2CCC(C1)N2C(=O)C(c1ccccc1)O c1(C(=O)NC2CN(C(Cc3cccc(C)c3)=O)CC2C)ccc(C#N)c(O)c1 CC(O)C(F)(F)C(=O)NCCN(C1CCCCC1)C(C1CC2CCC(C1)O2)=O c1(C(=O)NCC(CN(C)C(C2(c3ccno3)CCC2)=O)O)cncc2sccc12 C(=O)(C(CNC(c1c[nH]nc1Cl)=O)C(C)(C)C)N(CC(C(C)C)C)C C1(NC(c2c(Cl)cn(CC)n2)=O)CN(C(C2(C3CC3)CCC2)=O)CC2(CCC2)C1 Cc1cc(C)nc(SC2CCN(C(=O)CCC3CCCN3)CC2)n1.C(C(C)C)N Cc1cn2c(n1)CC(C(=O)NC1CC(NC(=O)C3=NOC(C)C3)C1)CC2 C1(C(=O)NCCC(C)NC(C2CC3CC3C2)=O)(COC)CCCC1 c1(NC(=O)NCc2nc(C(CC)C)on2)ccc(C)c(C(F)(F)F)c1 N1(C(Cc2c(C)n(C)cn2)=O)CCN(C(=O)CCCc2ccsc2)C2(CCC2)C1 C(CCCC(C)NC(=O)CN(C)CCO)NC(C(C)n1ccnc1)=O c1(C(N2CC(O)(C(C)NC(C(C=C)OC)=O)C2)=O)cc(CC)ccc1O N(C(=NCCO)NC1CCN(C(=O)CC(C)C)CC1)CC(=O)N(CCC)C(C)=O C12(C(=O)NC3C(NC(CC(CC)CC4CC4)=O)C3)CC3CC(C1)CC(CC)(C3)C2 C12(C(N(CCN(C(=O)CSC(F)F)C(C)C)C)=O)CC=CCN1CCC2 C(C(C(=O)N1CCCC1Cn1cc(CNS(C)(=O)=O)nn1)OC)OCC(=O)OC c1(CC)sc(-c2nc(CC(C)CC)nn2-c2ncnn2C)cc1C c1(C(=O)Nc2cccc(NC(C3C(COC)C3)=O)c2)cc(OC)cc(OC)c1 N1(C(CC(C2CC2)NC(=O)CC2CC3(CCC3)C2)=O)CCSCC1CO C1(OC)CC(CCNC(=O)CC(C)C)N(C(c2cncc(-c3cc[nH]n3)c2)=O)C1 C1(C(N2C(CNC(C(C(C)C)(C)C)=O)CCC2)=O)CCC2(CC1)CC2(F)F c1(NC(C2C(NC(C#CC(=O)O)=O)C2)=O)nccc2cc[nH]c12 Cc1ccc(CC(=O)NC2CC(C)(NC(C3CC3[N+](=O)[O-])=O)C2)cn1 CN1CCC(CC(=O)NC(Cc2cnc[nH]2)C(=O)NCC2C(C)(C)C2(F)F)CC1 c1(CC(=O)NC(CC)CNC(=O)C(C)CC)ccc(Cl)c(Cl)c1C C1(CC(N2CC3C(CN(C(c4c(C)nsc4C)=O)C)C3C2)=O)CCCCC(=O)N1 C1(NC(=O)C2=CCCSC2)CCC2(CCN(C(C3CCSC3)=O)C2)C1 C1(C(N2C3(CC(C#C)C3)CC2)=O)CCc2nnn(C3CCN(C)CC3)c2C1 c1(C2N(C(=O)C=Cc3ccsc3Br)CCC2)ccc(F)cc1Cl N1(C(c2cnc(C)c(N)c2)=O)CC2CN(C(C3CC=CCO3)=O)CC2C1 c1(C(=O)NC2CCC(NC(C3CN(CCC)C(=O)C3)=O)CC2)ccc(F)cc1Cl N1(C(C(CC)C2CCC(=O)N2)=O)CC(C2(NC(c3ncccc3C)=O)CC2)C1 C=CC1(C(=O)NC(C)C(=O)N(C)CC)CN(C(=O)CN2CC3CCC2C3)C1 N1(C(C=CC)=O)CC2CC(NC(C3CCC=CCCC3)=O)CC1C2 CC(C)C(C)C(CNC(=O)CC1(O)CCCCCC1)NC(C1CCC1)=O Cc1ccc(O)c(C(N2CCCC(CCNC(C3(CO)CC3(F)F)=O)C2)=O)n1 C(C(=O)N(C(C)CCNC(c1csc(CC)n1)=O)C)(C(C)C)SCC N1(C(C2CC(C(C)C)C2)=O)CCC2(CCCN2C(c2cccs2)=O)C1 c1(C(=O)Nc2ccc(SC)cc2)cnn2cc(-c3cccc(C(C)=O)c3)ccc12 N1(C(C)=O)CC(O)CC1C(N1CCCC1CN(C)C(C1C(C)C1C)=O)=O c1(NC)cc(Cl)ccc1C(N1CCC(CNC(c2cc(OC)cs2)=O)CC1)=O C1(C(N(CCC#C)C)=O)CC(NC(c2cnnc(O)c2)=O)C12CCC2 C1(NC(C=CC)=O)CCCC12CCN(C(c1ccc(NC(C)=O)cc1)=O)C2 CC1CC(NC(=O)CNC(=O)CCCF)CCN1C(=O)NCC(c1ccco1)=O C1(C(N(CCNC(c2c(C)nc(C3CC3)s2)=O)C2CC2)=O)CCC2CCCCN12 C(=O)(N=c1ccn(C)[nH]1)N1CCC(O)(c2cn(C(C)C)nn2)CC1 CCCCCC(C(=O)N(C)CCOCCN(C(=O)CC1=CCOCC1)C)C(C)C C1(C(=O)NC(CN2CCN(C(C3CC(SC)C3)=O)CC2)C)CCC2CC1C2(C)C c1(C(=O)NCC2C(NC(C(C)(O)C3CCC3)=O)CC2)cc(N)cnc1Br c1(C(=O)NCC2CCC(NC(C3(C(N)=O)CC3)=O)C2)nc(O)[nH]c(=O)n1 N1(C(C(C)OCCN(C)C)=O)CCC2(NC(=O)CCn3cccn3)CCCC12 N1(C(C2C3(CC3)C23CC3)=O)C(CNC(C2(CO)CCCO2)=O)CC2COCC12 CC1c2ccccc2CN1N(CC1CCCO1)Cc1ccccc1 CCCC(O)CC(=O)N1CC2CC1CN2C(c1cc(CN(C)C)on1)=O c1(C(=O)NC(CN(C(=O)C(O)Cc2cnc[nH]2)CC)C)cc(N)ccc1C CC1SCCN(C(=O)CCc2cccc(C#N)c2)C1C N1(C(C2C(C)CC2)=O)CCC2CC2(C(N2CC3(C=CCO3)C2)=O)CC1 Cc1cc(=N)[nH]cc1C(=O)NCC(CO)NC(=O)Cn1nc(O)ccc1=O C1(CCOC)CN(C(=O)COC2CCOC2)CCN1C(=O)C1CC1 C1(NC(CCCC(=O)OCC)=O)CC2CCCC(C1)N2C(=O)C(O)CC1CC1 c1(C(=O)NCC2N(C(c3cn4cc(C)sc4n3)=O)CC2)cnc2c(c1)CCCO2 c1(CCC(=O)NC2(CC(=O)N(CCC#C)CC)CCC2)cccnc1C c1(SCC)cccnc1C(N1CC(N(C)C(c2sccc2SC)=O)C(C)C1)=O N1(CC2C=CC(C(=O)OC(C)(C)C)C2)CCNC(=O)C1c1ccc(I)cc1 N1(C(c2ccn(CC)c2C)=O)CCCC(CNC(c2cc([N+](=O)[O-])c[nH]2)=O)CC1 C(=O)(N=c1cc(F)n(C)[nH]1)NC(CN(C)C)CCO C1(N(C)C)C2CN(C(c3ccc(OC(C)(C)C)cc3)=O)CC12 c1(NC(C2CCCN2Cc2cnc(C3CC3)s2)=O)cc(Cl)cc2ncoc12 C(CN=c1[nH]c(N2CCC(F)(CF)C2)nc2c(F)cccc12)N(C)C(=O)C1CC1 C1(CC(=O)NCCC(C)NC(C2N(CC)CCOC2)=O)CCc2ccccc2C1 c1(C(=O)NC(C)CCNC(C2(c3csc(Br)c3)CC2)=O)cncc(N)n1 Cc1cccc(C(N2CCC(CN(C)C(C34CC(CF)(CO3)C4)=O)C2)=O)c1 C1(CCNC(C2(NC(C)=O)CC2)=O)CCCN(C(C2CC2(C)C)=O)C1 N1(C(C2(CCCC)CCCC2)=O)C(CNC(=O)CC2CCC2)CC2CC12 C1(C(=O)NC)CN(Cc2cn(CC(=O)NCCOCCC=C)nn2)CCO1 N1(C(C(C(=O)OCC)CC)=O)CCN(C(c2cc(F)c(F)cc2F)=O)CC12CC2 C1(NC(C2C(OCC)C2)=O)CCC(CNC(c2cnn(CC)n2)=O)C1 CCC(C)CC(C)C(=O)NC1(CN(C)C(c2cccn(C3CCC3)c2=O)=O)CC1 c1(CC)cc(N(C)C(C2CCCN(C(C3CCC4(CC4)C3)=O)C2)=O)cc(C)c1 N1(C(c2c(CC)noc2)=O)CC(C)C(C)(CNC(C2(C)CC(C)(C)C2)=O)C1 Cc1cc(C(N2CC(C(=O)N(C)CC3CCCN3C)C(F)C2)=O)cnc1O N1(C(C2(OC)CCCC2)=O)CC(NC(=O)COCCN(C)C)C(C)C1 C1(C(=O)NC2CC(C)(C(N3CCC(CC(F)F)C3)=O)C2)CCCCC(=O)N1 O=C(NNc1ncnc2n[nH]cc12)c1ccc2ncccn12 CC1(CNC(C2CC2(F)F)=O)CCCN1C(=O)Cc1cccc(OCC#N)c1 CCC(CO)(C(=O)N1CC(OCCNC(=O)C(C)CO)C1)OC C1(CNC(C(C)CN(C)C)=O)CC(NC(=O)Cc2csc(Cl)c2)CC1O C1(C(N2CCN(C(c3nc(C)sc3)=O)CC2CCO)=O)CCS(=O)(=O)C1(C)C CC1CC(NC(=O)Cn2cccnc2=O)CN(C(=O)CNC(=O)CC(C)(C)C)C1 N1(Cc2c(C)ccc(O)c2)CCC2(CCCC2C(=O)Nc2ncco2)C1 c1(C(=O)NC2CC2)cccc(CNC(C2CNCCOC2)=O)c1 CC1(C(=O)NC2CCC(O)C2O)CCCN(C(=O)CC=Cc2ccccc2)C1 c1(NC(=O)NCC(CC=C)CO)cn2c(n1)CCCC2 CC1=C(C(=O)N2CCC(CNC(=O)CC(C)(C)O)C(C)C2)SCCO1 C1(C(N(CC(C)N(C(=O)CN2CCCNC2=O)C)C)=O)CC2(COCCO2)C1 C1(CNC(Cc2cccc(C)c2)=O)CC2CCC1N(C(=O)C(C)CC(C)(F)F)C2 c1(CC)ccc(C(=O)NC(C)CCCNC(c2ccnn2CC(F)F)=O)cc1 C(=O)(CCCN=[N+]=[N-])NC(CC(C)C)CNC(=O)C(C)(C)c1cscn1 C1(O)(C(=O)NCCC2CC(C(=O)Nc3cn(CC)nc3)C2)CCSCC1 C=CC(C)CC(=O)NC1CC(N(C(=O)CN2CC3CC3C2)C)C1 C1(C(C)(C)NC(=O)CSC(=N)N)CCCN1C(c1ccsc1C(=O)O)=O C(=O)(C(C(C)(C)C)OC)N(C)CC1C(NC(c2c(C)cns2)=O)CCC1 C1(NC(c2csc(Cl)n2)=O)COC2CN(C(c3ccc(CO)cc3F)=O)CC12 C1(C(N(C(C)CN(C)C)CC)=O)C2CC1N(C(=O)CC1(C)CCC1)C2 c1(CC(C(=O)OCC)NC(c2occ(C)c2C)=O)cn(C)nc1C c1(CN2CC(NC(c3ccc(C#N)c(Cl)c3)=O)C(F)C2)ccc2c(c1)CCCC2 C1(CNC(C2(CNC(C(C(C)O)NC(N)=O)=O)CC2)=O)CCOC2(CCC2)C1 Cc1cc(Cl)c(C(=O)N(CCC(C)NC(=O)Cn2ncccc2=O)C)cn1 c1(C(=O)NCCN(C(=O)Cn2c(-c3ccccc3)nnc2S)C)cc(F)n(C)n1 Cn1ccnc1CNC1CC(NC(c2ccc(C(C)(C)C)[nH]2)=O)C1 c1(OC)ccc(C(=O)Nc2ccc(CSc3ccccc3C)cc2)cc1N c1(C(N2C(CNC(=O)CCCn3cncn3)CCC2)=O)cccn2cnnc12 N#Cc1ccc(=NCCCNC(=O)CSc2ccncc2)[nH]n1 OC1(C2CCC2)CCN(Cc2nnc(-c3cccc(Cl)c3)o2)CC1 c1(CC)cncc(C(=O)NCCCC(C)NC(C2CCC(=O)NC2)=O)c1 C(CCN(C)C(c1cnc(O)s1)=O)(C(C)C)NC(c1ccn(CC(C)C)n1)=O N1(C(C2(c3c(C)cno3)CC2)=O)CCN(C(=O)C(=O)N(C)C)CC(O)C1 C1(C(=O)NC2CC(NC(C3(OC)CC3)=O)C2)CC2CC(=O)C1O2 CCCCC(CNC(=O)CCc1nc(C)c(C)o1)NC(c1cnc(NC)cn1)=O Cc1cc(O)ncc1C(=O)NCC1CCCCN1c1cc(O)ncn1 C=CCC(F)(F)C(=O)NCC(C)C(F)C(=O)NC1(C(O)COC)CC1 C(=O)(C1=COCCO1)OCCOc1cn(C2CN(Cn3c(C)ncc3)C2)nn1 C1(NC(C(C)C2CC2)=O)C2CC1N(C(C1CC(O)(C(F)(F)F)C1)=O)C2 C1(NCCCCCN(C(C(CC)NC(N)=O)=O)C)CC(OC)CN1C(C)=O Cc1nc2c(n1C)CN(c1nnnn1Cc1noc3c1CCCC3)CC2 Cc1cccc(OCC(=O)NCCC2CCN(C(c3csc(C)c3)=O)C2)c1 Nc1ccc2nc(N3CCC(NC(C4CC5C=CC4C5)=O)CC3)sc2c1 c1(OCC)cc(C(=O)NCCCOCCNC(=O)C(O)CSC)ccn1 c1(CNC2C(C)C(c3ccccc3)C2)cc(C2(C)CC2)ccc1F Nc1cc(Br)cnc1C(=O)NCC(CO)NC(C1CC2CC2C1)=O c1(SC)ncc(C(N2CCN(CCCNC3CC34CCNCC4)CC2)=O)c(Cl)n1 C1(NC(CCC)=O)CC2CC(NC(=O)C(O)COC)CC2C1 C#Cc1cncc(NC(C23CC(CN2C(c2ncncc2C)=O)C3)=O)c1 c1(N2C(C)CC(NC(=O)COC3CCOCC3)C2)nc(O)c2cnn(C)c2n1 N1(C(C(Cc2cccc(OC)c2)O)=O)CCCC(CO)(NC(C2(CO)CC2)=O)C1 c1(C(=O)NC(C)C(CO)NC(C2(C3CC3)CC2)=O)c[nH]c2c(Cl)cccc12 c1(C(N2CCN(C(CC(C)C(F)F)=O)CC2C(F)F)=O)cc2c(ncn2C)[nH]1 C(N=c1[nH]c2c(c(=NCCc3ccccc3CO)[nH]1)COC2)C1(S(N)(=O)=O)CC1 N1(C(c2n(CC)ccc2)=O)CC(NC(=O)CC23CCCC2C3)CC2(CC2)C1 C(=O)(C(CC)(CC)CC)C1OCCN(C(C(C(CC)O)C)=O)C1.C1CCN(C)CC1 N1(C(CC(C)F)=O)CCN(C(c2cc(Cl)sc2Cl)=O)C(CCO)C1 N1(C(CN(C)C(c2cscn2)=O)=O)CCC(CNC(C2CC3C=CC2O3)=O)CC1 c1(CC(=O)NCC2(CCNC(CCSC)=O)CC2)sc(C)nc1-c1ccccc1 Cc1cc(F)cc(CN2CC=CC2C(=O)Nc2csc3nccnc23)c1O Cc1ccc(C(=O)NCC2CC23CC3(F)F)c(O)c1Br N1(C(C2OCCC(NC(c3ncn(CC)c3)=O)C2)=O)CCC(F)(CO)CC1 c1(C(C)C)[nH]ncc1NC(C1CC1NC(=O)Cc1ccc(Cl)s1)=O c1(CC(CNC2C(C)SCC2)O)ccc(C(F)(F)F)cc1 C1(C(=O)NCC(CC)NC(C2(F)CCOCC2)=O)Oc2ccccc2OC1C C1(Cc2nccc(OC)c2)CN(C(=O)COC2CC2C(=O)NC)C2(CCC2)C1 CCC(CC)(CO)C(=O)N1CC(F)CC1CC(N1CCC(CC(N)=O)C1)=O CC1CN(C(=O)CCC#N)CCC1N(C(=O)COC1CCCCCC1)C c1(NC2CN(C(CCCC#C)=O)CC(C)(C)C2)nc(C)nc2scc(C)c12 C1(NC(C(CC)SC)=O)CN(C(c2cnsc2C)=O)C2(CCCCC2)C1 C(=O)(C1=NN(CCO)C(=O)CC1)NCC1CN(C(C(COC)O)=O)CC(C)(C)O1 C#Cc1ccc(C(=O)NCC2CC2NC(C2CC3CC3C2)=O)c(F)c1 N(C(=NCCc1ccccc1F)N1CCSC2(CCCCC2)C1)C(COC)C c1(CN2C(CCC(=O)NC3CC3(F)F)CCC2)cc(F)c(F)c(Cl)c1F C(=O)(C1=CC2C=CC1C2)N1CC(OCC(N)=O)C1 N1(CC)CCCC(C(=O)NC(C)CCN(C(=O)CCc2ccc(C)cc2)C)C1 N1(S(CC(CC(C)C)OC)(=O)=O)CC(C(=O)OC)CC(C)(C)C1 c1(C(=O)NC2(c3ccc(-c4cn(C)nc4)cc3)CCC2)ccc(O)cc1F c1(CC(=O)NCC2N(C(c3c(CC)nc[nH]3)=O)CC2)c[nH]c2cccc(OC)c12 CC(C)=C=CC(=O)NCC(c1ccccc1)CNC(=O)C=CBr C1(NC(CC(CC)SC)=O)CN(C(c2ccc(-c3ccco3)[nH]2)=O)C2(CCC2)C1 c1(C(=O)NCC(C)CNC(=O)C(C)n2cccn2)cc(C(F)(F)F)ccc1O c1(C(=O)NC2C3CN(C(c4n(C)ncc4)=O)CC32)ccnc(F)c1F c1(NC(CNC(CC)=O)=O)cn(C)c(C(=O)NCc2ccc(C(=O)O)o2)n1 CCC(C)C(=O)C(=O)NC1CC=CCC1C(N1CCCCC1C(=O)NC)=O N1(C(C2(C)CC(F)C2)=O)CC(NC(=O)CNC(N)=O)CC2(CCC2)C1 CC1C(NC(=O)C(F)(F)c2nccs2)CC2CCC1N2C(c1cncc(Cl)n1)=O c1(C(N2CC(NC(C3CC(CC)OCC3)=O)(CO)C2)=O)n[nH]c2ccc(F)cc12 N1(C(=O)Cc2ccoc2)CCCC(C2CCCN2C(c2cc(C3CC3)no2)=O)C1 CC(C(C)(C)C(=O)NCC1CNC(=O)C1)NC(=O)CC1CCOC1=O CCCC(CCC)CC(=O)N(C)CC1CCCN1C(=O)Cc1cc[nH]n1 c1(OCC(=O)OC)cc2ccccc2cc1NC(=O)C#CC1CCCC1 CCCCCC(C)(C)C(=O)NCCN(C(=O)CCC1CCCCN1C)CCC N1(C(C(c2cccc(C)c2)O)=O)C2CCC1CN(C(C1CC3CCC1C3)=O)CC2 c1(C(=O)NCC(C)NC(C2CSCC(=O)N2)=O)cc(N)cc2c1OCCO2 c1(C(=O)NCC2(O)CN(C(=O)C(F)(F)c3csc(Cl)c3)C2)cccc2nncn12 c1(C(N2CCC(OC)(CNC(=O)C=C3CCC3)C2)=O)cccc2nc(O)[nH]c12 C12(COC)CC(NC(C3(C)CCOC3)=O)(CN1C(c1cccnc1N)=O)C2 C1(C(=O)NC2C(C)CCN(C(CN(CCC)C)=O)C2)CCS(=O)(=O)C(C)C1 C(C(C)C(C)n1cc(Cn2cnc(CO)c2)nn1)OC Cc1nn(CC(C)C)c(Cl)c1C(=O)NCC1(CCNCCN2CCCC2)CC1 N1(CC)CCOC(C(N2CC(CCN(C(=O)CC3C=CCC3)CC)C2)=O)C1 c1(C(=O)NCc2cn(CC3CCCCNC3=O)nn2)ccc2c(c1)S(=O)(=O)NC2 c1(N2CC(C)N(C)C(=O)C2)nc(=NCC2(N(C)CCO)CC2)[nH]c2cc[nH]c12 c1(C(N(CC(C)N(C(c2sc(C)c(C)c2C)=O)C)C)=O)ccc(F)c(F)c1N Cc1cccc2cc(C(=O)NC3CC(C)N(C(c4cnn(C5CC5)c4)=O)C3)[nH]c12 CCCCCCCC(F)C(=O)NCCC(C)NC(=O)CC12CCCC1C2 N1(C(CCc2cn(C)nc2)=O)CCC2(NC(=O)CCc3cocn3)CC2C1 N1(c2nccc(C(=O)Nc3ccc(F)cc3)c2)CCn2cccc2C12CCC2 c1(CC2(C(=O)NCCC(C)N(C(c3cc(C)ns3)=O)C)CC2)c(F)cccc1F C1(OC)CCCN(C(C2(C)CCN(C(C3COCC3C(N)=O)=O)C2)=O)C1 C1(F)(C(=O)NCCC2OCCN(C(C3COC3)=O)C2)CCS(=O)(=O)C1 C1(NC(C(C)OCC=C)=O)CCC(NC(c2ncc(C(F)(F)F)s2)=O)CC1 CC1CN(C(C2C(Cl)(Cl)C23CC3)=O)CC2(CCN(C(=O)C(C)(C)C(F)F)CC2)O1 CC(C)C(F)C(=O)N1CC=CC(NC(=O)CCN(C)CCO)C1 c1(SC)cccnc1C(N1CCCC(CCNC(=O)Cc2cncs2)C1)=O C1(Cc2cn(CC)nn2)(C)CCCCCC1.C(=O)C(CC)CO Cc1cc(F)ccc1NC(=O)C(N1CCC(CC2CC2)CC1)c1cc(C(F)F)no1 N#Cc1ccc(NC(c2cncc(-c3cccc(C4(C#N)CC4)c3)n2)=O)c(I)c1 CC(C)CC(O)C(C)C(=O)N1C2CCC1C(C(=O)Nc1cncc(CO)c1)C2 c1(C(N(CC(CC)NC(c2cnc(O)o2)=O)C)=O)cnc2cc(C)ccn12 CN1CCCC1C(=O)NCC1(C(N2CC(CC(F)F)C2)=O)CCCC1 Cc1cc(S(=O)(=O)NC2CCN(C)C(=O)C2)cc(Br)c1C CCCCC(F)C(=O)NCC1(C(=O)NCCCc2cncnc2)CC2(CC2)C1 CN1CC2(CCN(c3nc(=N)[nH]c(=NCc4nc(C(N)=O)co4)[nH]3)C2)CC1=O c1(C(=O)NC(C(C)NC(C2(C)CCOC2)=O)CO)c(N)cc(F)cc1F c1(CC)oc(C(=O)OCCc2ccc(F)nc2)cc1C(=O)NC C(=O)(C(C)C(O)CC(C)C)NC(C(N1CC=C(COC)CC1)=O)Cn1cccn1 c1(CN2C(C(N3CCCC3c3ccc(Cl)s3)=O)CC(O)C2)ccc2ncnn2c1 N1(C(Cc2ccn(CC(C)C)n2)=O)CCC(NC(=O)CC#N)C(C(C)C)C1 c1(C(=O)OC(C(=O)NCC2C(C)C2)C)cccc(C(=O)OC2CC2)c1 c1(C(=O)NC2CN(C(c3c(CC)n(C4CCCC4)nc3)=O)C2)ccc(F)c(F)c1 C1(C(=O)NC(CN(C(c2ccnc3ncnn23)=O)CC)C)Cc2nnc(C)n2C1 C(CCCCO)N(C)C.C12CC(C1)C(=O)NC2.C12CC(C1)CC(=O)N2.C(C)(=O)O C(=O)(C1=C(Cl)CCOC1)N(CC(C)O)CCNC(=O)C(O)CC(N)=O CCCCCC(F)C(=O)N1CC2C(C(=O)NOCC(O)C(C)C)C2C1 c1(C(=O)NC2CN(C(c3c(CC)non3)=O)CC2C)cc(C(F)(F)F)ccc1F C(=O)(CC1CC(=O)Nc2ccccc21)N1CCC(C)(NC(C2CCCC2)=O)C1 N1(C(CSCCC)=O)CCC(C)(CNC(C2(CC(C)C)CCNC2=O)=O)C1 CC(C)C(C)(Br)C(=O)N(C1CN(Cc2ccccc2)C1)C S(=O)(=O)(c1ccc(C)cc1)NCC(=O)NCC(CC=C)NC(=O)CC(C)C=C N1(C(Cc2cc(C)no2)=O)CCC2(NC(C3(CN4CCCCC4)CC3)=O)CCCC12 C(C(C(=O)N=c1cc(C)n(CCO)[nH]1)NC(c1cnsn1)=O)SCC c1(C(=O)NC(C(CO)NC(c2c(CC)onc2C)=O)C)ccc2ncsc2c1 c1(C(=O)NC2C(NC(C3CCN(C(=O)NC)CC3)=O)CCCC2)ccc(F)c(Cl)c1 CCC(C)(O)C(=O)N1CCCC(NC(c2ccccc2Cc2nc[nH]n2)=O)C1 C1(C(N(CCNC(CCn2ncc(C)c2)=O)C)=O)CCC(C)NC1=O c1(OC)ncnc(OC)c1C(=O)NC1CN(C(=O)CCCN(C)C(C)C)CCC1C Cc1cnc(C(=O)NC(C)(C)CN(C(=O)C(C)n2cnnn2)C)cc1C N1(C(C2CCCOC2)=O)CC(C2CC2)(C(=O)NCCCc2cccs2)C1 Cc1cccc(C(=O)NC2(C(=O)NCC(F)(F)C(C)C)CCN(C)C2)c1F C1(NC(c2nc(CCC)sc2)=O)CCN(C(C2CC(F)(CO)C2)=O)C(C)C1 c1(CCc2nc(-c3cn(C)nc3)nn2C2CCS(=O)(=O)C2)cc(F)cc(F)c1 C1(N(C(=O)CCc2csc(=N)[nH]2)C)CN(C(C2(CF)CCOCC2)=O)CC1(C)C C(=O)(C1CCCc2ncnn21)NCC1(O)CCN(C(c2c(F)ccc(C)n2)=O)C1 c1(NC2(Br)C(C)C2C)c(C(N)=O)cccc1C(=O)O N1(C(C(CC)=CC)=O)CCC2CCCC12CNC(=O)Cc1ccc(C)c(C)c1 C1(OCCC(=O)NC(CC2(C(=O)OC)CC2)=O)COCCC1OC1CCCCC1 C1(OC)CC(CO)N(C(=O)CC2CCN(C(=O)C(c3cnccn3)C)C2)C1 c1(C(N(C2CN(C(C(C)O)=O)CC2(C)C)C)=O)ccnc2c(Br)cccc12 n1(CCC)cc(C(=O)NC(C2CN(C(C3(C4CC4)CCCO3)=O)C2)C)nn1 c1(C(N2C(C(=O)NCc3cc(C)no3)C(C)CC2)=O)cccc(=O)n1C c1(C(=O)Nc2c(-c3n(C)ncn3)cc(Cl)cc2)c(N)cc(F)cc1F c1(NC(C)=O)ccc(OCC(N2CCOCC2CNC(=O)C(=O)N(C)C)=O)cc1 c1(C(=O)NC2C(CNC(C(CC)N(C)C)=O)CC2)ccc2cc[nH]c2c1 N1(C(c2n(CC)nnc2)=O)CCC(NC(=O)CCn2cccnc2=O)CC(O)C1 c1(C(N(c2ccc(F)cc2)CCCC#C)=O)ccc(I)c(C)c1 c1(C(=O)NC(C(=O)NCc2c(C)csc2)C2CCCO2)cccc2ccnn12 c1(OC)nccc(C(=O)NCC2(F)CC(CNC(=O)CSC(F)(F)F)C2)c1F C1(OCc2c(C(=O)OC)nco2)(CN)CCCCC1.C1C(C)NC(=O)N1 c1(C(N2CCC(C)(CNC(C3CCCCS3)=O)C2)=O)cccc(NC(C)=O)c1 C1(C(N(C(C)CNC(=O)CCN2CCCC2=O)C)=O)CCC2(CCC2)OC1 C(=O)(C(C)(C)C(F)(F)F)N1CCCC(NC(c2nccc(C)c2N)=O)CC1 C(=O)(NNc1cccc(C(C)C)c1)C1(Cc2ccc(C)cc2)CCCC1 N1(C(CC(CC)C2CC2)=O)CC(C(=O)NC2(C)CC(F)(F)C2)C2(CC2)C1 C(=O)(C1=CS(=O)CCC1)NC(CNC(c1cnc(OC)c(C)c1)=O)CC(F)(F)F c1(NC(C2N(C(=O)NC(C(=O)OC)C)CC(O)C2)=O)cnc(Cl)c(Br)c1C CC1CC(NC(C2(CC(F)(F)F)CC2)=O)CN1C(c1ccc(C2CC2)cc1)=O CS(=O)(=O)CCCC(=O)N1CCC(CCNC(C2CC(C(F)(F)F)C2)=O)CC1 c1(C(=O)NC(C)CCNC(C2CC(F)(CO)C2)=O)ccc(N)c(F)n1 c1(CCC)c(C(=O)NC(C2(O)CN(C(c3cc[nH]c3C)=O)C2)C)nnn1C c1(CNC(CN(CC)CC)=O)cccnc1CNC(=O)C=C(C)C C1(Cl)(C(=O)NCC2(O)CCCN(C(c3cn(C)nc3Cl)=O)C2)CC12CCOCC2 C1(C)(CNC(c2cnc(OC)s2)=O)CCN(C(=O)CCC(=O)N2CCOCC2)C1 c1(C(N2CC(NC(c3ccc(Br)o3)=O)C(F)C2)=O)ccc2c(n1)CCCN2 C1(N(C(c2c(CC)ncs2)=O)C)CCCC(N(C(=O)CCc2nccs2)C)C1 N1(C(C(=O)NCc2ccc(OCC)cc2)=O)CCCC(F)(C(=O)O)C1 CCCC(c1nnnn1CC1CCCO1)(C1CCCCC1)NCc1cocn1 CC1(C)C(NC(c2ncoc2C(=O)O)=O)CC1CNC(=O)CC1(C)CCOCC1 C1(NC(C(C=CC)O)=O)CC2(CCN(C(=O)C(C)(F)CCCC)CC2)C1 c1(OC)cn2c(cc1=O)CN(C(=O)CCc1ccc(S(N)(=O)=O)cc1)CC2 C1(O)(CCNC(CCC=C(C)C)=O)CCN(C(c2ccnc(O)c2)=O)C1 C(C(=O)N=S(C)(=O)c1cnn2c1CN(C(=O)C(C)(O)C1CCC1)CC2)=CC N1(C(c2ccc(C(CC)=O)cc2)=O)CC(C)C(NC(c2cc(C)cs2)=O)C(C)C1 N1(C(CCCOCC)=O)CC(NC(C2CCCS2(=O)=O)=O)C(C(F)F)C1 N1(C(N2c3ccc(OC)cc3OCC2)=O)Cc2c(ccc(F)c2Br)CC1C C(=O)(C(F)(F)C(C)O)N(C(C)C(=O)NCc1cccc(F)n1)CCC c1(C(N(C(CN(C(C(C)N(C)C)=O)C)C)C)=O)cc2ccc(Br)nc2[nH]1 c1(-n2cc(CC(C)C)nn2)ccccc1OCCN(C)C.C12(CC1(F)F)C(=O)N2 c1(N(C(C(=O)NCCOCCN(C(COCCCC)=O)C)=O)C)ccc(CO)o1 N1(C(=O)Nc2cc(C)cc(C#N)c2)c2ccccc2CC1C C1(CN(C(C(C)OCCC=C)=O)C)COCCN1C(=O)Cc1ccsc1 C#Cc1cccc(OCC(N2CC(CC(C)(C)CNC(=O)C(=O)NCC)C2)=O)c1 c1(CC)nccn1CCNC(=O)C(CN(C)C)NC(c1cnn[nH]1)=O C1(C2CCCCO2)(C(=O)NOC2CNC2)CCCO1 C1(C(=O)NC(C2(OC)CCC2)C)CC(=O)CN1C(C1CNC(=O)N1)=O C1(CNC(C)=O)CN(C(C2C(F)(F)C23CC3)=O)CC2(CCC2)O1 c1(-c2ccc(C#N)cc2)n[nH]c(=NC(=O)NC(C2CC=CCC2)C2CC2)s1 c1(C(C)C)nn(C)cc1C(N1CCC(C)(NC(=O)CC(C)c2cccnc2)C1)=O C(N=c1[nH]c(CC)nc(Cl)c1CC)C1(C)CCC(NC(C(F)=CCC)=O)CC1 O=C(C1=NOC2(CCC2)C1)NC1C=CCCC1C(=O)NCC1(O)CC1 c1(C(=O)NC(CC(C)NC(CCS(=O)(=O)NC)=O)C)n[nH]c2c1CN(C)CC2 c1(CC)c(OC)cccc1C(=O)NC1CC1NC(=O)C(C)Cc1cnn(C)c1 C1(CC(=O)NC2CN(C(Cc3nc(C)oc3)=O)CC(F)C2)CCn2cncc2C1 C(=O)(C(C)(CC)C(F)F)NCC(c1cccc(C)c1)NC(c1c(CC)n[nH]c1)=O C(=O)(C(C)(C)C(=O)N1CCCC(CCCCNC(=O)CCC(N)=O)C1)N(C)C C1(NC(C2CC(OC)(OC)C2)=O)COCCN(C(C2CC3CCC(C2)S3)=O)C1 Cc1ccc(C(N2CCN(C(C3CC3C3CC3)=O)C(C3CC3)C2)=O)c2c1CCC2 CCCC(C)(C)CC(=O)N1CC2CC(C(N3C4CCC3COC4)=O)(C2)C1 CCC(CC(F)F)C(=O)NC1CCCC1NC(c1cnc(C)c(C(C)=O)c1)=O N1(C(=O)C=CSc2ccccc2)CCCC(CNC(C2(O)CC2)=O)C1 c1(C(N2CCC(CNC(C(CSC)OC)=O)C2)=O)cc(C)c(C)nc1O N1(C(C2(NC(c3occ(C)c3)=O)CCC2)=O)CCCC(F)(CO)C1 c1(NC(c2cccc(OC)c2)CNC(=O)OC(C)(C)C)cnc(C)c(C)c1C C(=O)(C(C(C)(C)O)CNC(=O)CN(C)C)NC(c1nc(CC)on1)C Cc1ccc(C(=O)N(CCC(C)NC(=O)C(C)(C)c2cnco2)C)cc1Br c1(OC)cc(C(=O)NCC2CN(C(C3COCCO3)=O)CCO2)cc(F)c1C#N n1(CC)cnc2nc(N3CCC(C4CC4)CC3)nc(N3CC4NC(=O)OC4C3)c12 c1(C(CO)N(CC(C)C)C(=O)NCc2nn[nH]n2)ccc(Br)cc1 C1(C(=O)NCC(CSC)OC)CC=CCN1C(c1ccc(CO)cc1)=O C=C(Cl)CCC(=O)NCC1CCC1NC(C1(C(=O)NC)CC1)=O C(=O)(C(F)(F)C(C)(C)O)NCC(CNC(C1C(C)OC(=O)N1)=O)(C)F C(CCC(C)C(=O)N(CC(=O)NCCCCc1cnc[nH]1)C1CC1)OC C(=O)(C(C)CCCC(C)C)NC(C(C)NC(CCC(=O)OCC)=O)C N1(C(CC2CCC(C)CO2)=O)CCC(F)(CNC(=O)COCC2CCC2)CC1 C1(C(N2CC(CNC(=O)CSCc3ccc(Cl)s3)C2)=O)Cc2ccccc2CO1 C(C(C(=O)NCC(C)N(C)C)NC(c1cc(CCC)[nH]n1)=O)SCC.N(C)C Cc1ccc2c(c1)C1CN(C)CCC1N2C(=O)OC(C)(C)C CC(C)(C)CC(O)CNC(C1C=CCN(C(c2cccnn2)=O)C1)=O c1(C(N2CCC(CC(=O)NCC(C(C)O)C)C2)=O)ncc(Br)cc1Br Cc1c(O)ccc(C(=O)NC2(C)CC(NC(C3CCCNC3=O)=O)C2)c1C CC(C(=O)NCCn1cc(C(N2CCC2C2CCOCC2)=O)nn1)C(F)F CC1CN(N2CC3(CC(Oc4ccccc4)C3)C2)CC(C)(C)O1 c1(C(N2CCCC(C)(NC(CNC(C(CC)C)=O)=O)C2)=O)cn2cc(C)nc2s1 C1(C(=O)NCCNC(C(CCC)OC)=O)(COC)CCCNS1(=O)=O C1(CNC(CCOCCOC)=O)CCN(C(=O)CSc2cccc[n+]2[O-])C(C)C1 N1(CCC)CCCN(C(=O)CC2(NC(c3ccsc3C#N)=O)CCCCC2)CC1 C(C1CCCC1)=C(C)C(=O)NCCCCCN(C)C(c1sccc1F)=O c1(C(C(N2CC(NC(c3n[nH]c(C)c3F)=O)C(O)C2)=O)O)ccc([N+](=O)[O-])cc1 C#CCC(C(=O)N1CCC(CCNC(c2cnc(C(C)(F)F)s2)=O)CC1)C1CC1 CC1(C)CCN2C(C1)C2=O.C1(NC=O)CC=C(C(=O)N2CCCC2CF)C1 C1(=O)C(CCSC)Nc2c(ncs2)N1CC.NC.OC Cc1ccc(C)c(Cn2cc(CCCNC(c3ocnc3C)=O)nn2)c1 C1(NC(c2c(CC)cno2)=O)COC2CN(C(=O)C(F)(F)C(C)O)CC12 N1(C(CCSC)=O)CC(NC(=O)C(C2(O)CCCC2)F)CC(C)(C)C1 C(=O)(C(C)(C)CF)N(CC(CN(C)C(c1c[nH]nc1-c1ccccc1)=O)O)C C12(CNC(c3csc(Cl)c3)=O)CC1CN(C(=O)CCCc1ccncc1)C2 N1(C(CCCSC)=O)CCN(C(=O)C2=COCCO2)C2CCC12 c1(NC(=O)CC(F)(F)F)ccc(S(=O)(=O)NC2CCCc3ccoc32)cc1F c1(C(=O)NC2(C(N(CC3=CCCOC3)C)=O)CC2(C)C)cnc2n1CCC2 C(C(CC(C)C)C(=O)NCc1nnn(C)c1C(N1CC(C#N)C1)=O)OC C1(NC(=O)CNS(=O)(=O)C2CC2)CCN(C(=O)CCC2NC(=O)NC2=O)CC1O C1(CNC(=O)CCF)CN(C(c2cccnc2Oc2ccc(Cl)cc2)=O)CCO1 C(=O)(CCC(F)(F)F)N1C(C(=O)NCCCP(C)(C)=O)C(O)CC1 N1(C(c2ccc(Cl)cc2)=O)CCc2sc(-c3cccn3-c3ccccn3)nc2C1 CC1=C(C(=O)N2CC(F)(CNC(c3ccc(C(C)(C)C)nc3)=O)C2)CCO1 c1(OCC(=O)NCC(C)N(C(=O)C=CC(=O)N(C)C)CC)nc(O)nc(O)n1 C(=O)(CCCC(=O)N1CCC(C(C)Nc2nc(C(F)(F)F)cc(C)n2)C1)NC c1(CC(=O)NCC(C(C)C)NC(C(C2CCCCC2)OC)=O)ccc(F)c(F)c1 c1(OC)ccccc1Nc1cscc1C(=O)NC1CCC1COC.C12CCN1C2 c1(C(N2CC3(CCN(C(C4C5CCC45)=O)CC3)C2)=O)ccc2ccccc2c1 Cc1nc(SC(F)F)sc1CC(N1CC(NC(c2c[nH]c(C#N)c2)=O)CC1C)=O C=C(C)C(C)(C)C(=O)N1CCN(C(=O)COc2ccc(F)cc2O)C(C(F)F)C1 CC1CCC(CC(=O)N(C)CCN(C)C(c2occc2Br)=O)C1 C1(CC=C)(NC(c2cc(-c3ccncc3)no2)=O)CN(C(C2CC(F)C2)=O)C1 Cc1ccnc2c(C(=O)NC3C4CC3CN(C(=O)C(C)S(N)(=O)=O)C4)cnn12 N1(C(c2[nH]cc(C#N)c2)=O)C2CCC1CN(C(c1cc3ccccc3[nH]1)=O)C2 C(c1cncc(OC)c1)=CC(=O)N(CCN1CCN(C(C2(C#C)CC2)=O)CC1)C N1(C(C(CSC)OC)=O)C2CC1CN(C(=O)CC1(C)CCOC1)C2 CC1CN(C(=O)C=C(C2CC2)C2CC2)CC(C)CN1C(c1c[nH]cc1Br)=O c1(OC)ccc(CNC2CN(c3ncc(I)cn3)CC2C)c(Cl)n1 N1(C(C(COC)O)=O)CC2(CCCC2NC(=O)C=Cc2cc(C)cc(C)c2)C1 N1(C(c2ccc(NC)cc2)=O)CCC2(NC(=O)CN3CCS(=O)(=O)CC3)CC2C1 CC(CCC(=O)N(C)CC1CCCN1C(c1ccncn1)=O)N(C)C Cc1ccc(Br)nc1CNC(N1CCCC(C)(F)C1)=O c1(CN2C(C(=O)NC(c3ccncc3)C)CC3(CC3)C2)cc(F)c(Cl)c(Cl)c1 c1(C(N2C(C(C(=O)NCC3CCN(C)C3)(C)C)CCC2)=O)nccc2[nH]ccc12 N1(C(c2c(CCC)[nH]cc2)=O)CC2(C=C(C(=O)NC(c3scnc3C)C)CO2)C1 CC1Oc2ccccc2N(CCC(=O)NCCc2cccs2)C1=O C1(NC(CC2(CC)CCC2)=O)CC(NC(C2CC3(C2)CC(C)C3)=O)C12CCC2 c1(OC)cc(Cl)c(C(N2CCC2CNC(C2CC(=O)NC(=O)N2)=O)=O)cc1Cl C(=O)(C(C)(C)C(=O)N1CCC(C)(CCNC(=O)CCN(C)CCO)C1)OC N1(CC(=O)NC(C(C)C)C)CC2CCC1C1CN(C(=O)Cc3ccn(C)n3)CC21 c1(C2SCC(NC3(CC=C)CCNC3)C2)ccc(F)cc1 c1(OC)ccc(CSC2CCCCOC2)cc1S(=O)(=O)NC(C)CC(C)N CCCCCCCC(=O)NC(C)CC(C)NC(=O)Cc1cc(F)ccc1F CC(c1cccs1)=CC(=O)NCC1CC1CNC(=O)CC1(C)CCOC1 C(=O)(C(=O)N=c1c(I)c[nH]cc1I)NCC(CC)CO c1(C(N2C(CCNC(C(C)n3cncn3)=O)COCC2)=O)cc2cc(Cl)sc2[nH]1 CC1CN(C(=O)CNc2ccc(Cl)cc2)CCCN1C(=O)CN(C)C(=O)C1CC1 C(=O)(CS(=O)(=O)C(C)(C)C)N1CCCCCC(NC(CC2CC(OCC)C2)=O)C1 c1(OC)ccc(Cl)cc1C(c1nnnn1C(C)C)NC1CCOCC1F C(=O)(C(F)C(C)C(F)(F)F)N(C1CCN(C(c2nc(O)c(C)s2)=O)C1)CC S(=O)(=O)(c1cc(Cl)c(O)c(Cl)c1)Nc1cccc(COC(C)(C)C)c1 N1(C(C(COC)(C)OC)=O)CCN(c2ccc(C(=O)NCC3CC3C)cn2)CC1 CC1CN(C(=O)C=C2CCOCC2)CC(CCNC(c2cc(=O)n(C)cn2)=O)O1 c1(C(=O)NCCC2(C)CN(C(=O)OC(C)(C)C)C2)cnc2ncccn12 N1(C(C2CC(=C)C2)=O)CC(CO)C2(CCN(C(=O)Cc3ccc(F)cc3)CC2)C1 N1(CCCCN)CCNC(=O)C1CCCl C(=O)(C(C)S(N)(=O)=O)N(C1CCN(C(=O)Cc2cnc(C)o2)CC1)CC#C C(C1=NOC2CCCC12)NC(CCN(C(Cc1c(C)ncs1)=O)C1CC1)=O C1(C(=O)NC2(CNC(c3cn(CC(N)=O)nn3)=O)CC2)CCC(F)(F)CO1 c1(CCC(N2C(C)CC(NC(c3cc(Cl)cs3)=O)C2)=O)c[nH]c2ccccc12 CC1CC=C(C(=O)N2CCN(C(c3ccc4nc[nH]c4n3)=O)CC2)CC1 c1(C(N2C(CNC(=O)C=Cc3cccc(F)c3)CCC2)=O)ccc2c[nH]nc2n1 Cc1cccnc1C=CC(=O)NC1(CNC(C2(N(C)C)CC2)=O)CCC1 N1(C(C(C(CC)O)C)=O)CCC2(CC1)CN(C(=O)CC1CCC(=O)C1)CCO2 C1(NC(CNC(CC)=O)=O)CC(O)CN(C(=O)Cc2csnn2)C1 N1(C(CC(CC)CN(C)C)=O)CC(NC(=O)CCc2ccsc2)CC(F)(F)C1 N1(C(CCCOCC)=O)CC2CC(NC(c3cnccc3OC)=O)C(C2)C1 CC1CCN(C(=O)C2=CCCS2)CC1CNC(=O)CC1OCCC1(C)C C1(CNC(C(CC=CCC)C)=O)CC2(CO1)CN(C(=O)CC(C)(C)C1CC1)C2 NS(=O)(=O)c1cc(C(N2CCC2CNC(C2C=CCC2)=O)=O)ccc1Cl C(CC(C(F)F)c1ccon1)NC1CC(C(N(C)C)=O)C1 C1(=CC(=O)N(CCCNC(c2cscc2F)=O)CC)CCCCC1(C)C C1(CC(=O)NCCN(C(CCCC)=O)C2CC2)COCC1(C)C Cc1ccc(C(N2CC3C=CC2C(C(N2CC(C)C(C)C2C)=O)C3)=O)cc1C#N C1(CC)(CC)CC(NC(=O)C(C)(C)N=[N+]=[N-])CN1C(c1csc(Cl)n1)=O c1(CNC(C2CC(=C)C2)=O)ccc(C(=O)NC(C)C(C)C(=O)OC)cc1 c1(CNC(C(N2CC(CC)(CC)OCC2)=O)=O)ccc([N+](=O)[O-])cc1Br.O C(CN=c1cc(-c2ccccn2)nc(Cl)[nH]1)c1cncc(OC)c1 CC1CC(NC(c2ccn(-c3ccccc3)n2)=O)CN1C(C1CC=CC1)=O C(=O)(C1=CCC2CCC1N2C(=O)CCc1cc(C)[nH]n1)NC1C(OC)CCC1 c1(CC(=O)NCC(CNC(=O)C(C)Oc2ccccc2)OC)c(C)cnn1C C(=O)(CCC(C)=O)NCCCNC(C(C)OCC#C)=O CC(C)(C)CC(=O)NCC(CC(=O)N1CCCCC1C1CC1)C1CCC1 C1(NC(c2cnc(OC)c(F)c2)=O)CCN(C(c2nocc2Cl)=O)CCC1CO C(N=c1ccnc(N2CCC(C3CC3)CC2)[nH]1)c1ccc(N(C)CC2CC2)cc1 C(c1cccc(F)c1)=CC(N1CCC(O)(CNC(C2(CC(C)C)COC2)=O)C1)=O C12(CNC(CCC(C)SC)=O)CCCC(CN1C(=O)C=Cc1cnccc1C)C2 c1(C(N2CCCC(N(C(C(CCC)C)=O)CC)C2)=O)[nH]c(C)c([N+](=O)[O-])c1C Cc1ncc(CC(=O)NC2CCC2CNC(C2(CS(N)(=O)=O)COC2)=O)o1 N1(C(=O)CC2CC(F)(F)C2)CCC(CCCN2CCNCC2)CC1 C1(C(N2CC(CNC(CC(CC)O)=O)N(C)CC2)=O)CCC2(CC1)CC2(F)F N1(C(CCc2n(C)ccc2)=O)CCC2(CC1)CC2C(=O)NC(CCO)C(C)(C)O C(CCc1ccc(Cl)cc1)(C(C)(C)C)NC(=O)NCC1OCC(C)C1 C1(NC(C2(CCOC)CCCC2)=O)CC12CCN(C(=O)CCCCC(C)C)CC2 CN1N=C(CC(=O)NCC2CC(F)CN2C(C2CC=CCC2)=O)CC1=O c1(C(=O)OC(C)C(=O)Nc2cccc(CCCC)c2)ccc(OC)c(C)c1 N1(CC(=O)NC2CCC(F)(CNC(CCNC(=O)OC)=O)C2)CCP(C)(=O)CC1 C12(NC(CN(C)C(N)=O)=O)CC3CCC(C1C2)N3C(C1CC(S(C)(=O)=O)C1)=O CC(CC(=O)NC1C2CC1CN(C(C1CC3(CCC3O)C1)=O)C2)C(F)F C12CCCCC1CC1CN(C1)C2=O.c1(OC)cnc(C(C)C)o1 Cc1cncc(C(=O)NCCC2CCN(C(c3ccon3)=O)C2)c1C c1(C(=O)NC2C=CCC(C(=O)NCC#CCOC)C2)ccc(C#N)c(C)c1 c1(SCC(=O)NCC(CC)NC(=O)C(F)C2CCCC2)nncn1C(C)C C12(C(=O)NCC3N(C(COCCOC)=O)CC(OC)C3)CCC(F)C1CC2 C1(C(N2CCC(CCF)CC2)=O)(OC)CCN(C(=O)C(=C2CCCCC2)F)C1 N1(C(C2C(C)(C)CCN2C(=O)CC2CCCO2)=O)CC2(CCCCCC2)C1 C=CC1CN(C(=O)C(F)(F)CN(C)C)CC1NC(=O)CC1CSCCS1 C1(NC(CC2(CC=C)CCCC2)=O)C2CCN(C(C3CCCCO3)=O)C12 C=CCCC(C(=O)NCCCCOC)NC(=O)CCC1CC1C C1(NC(C(c2ccc(OC)cc2)O)=O)CC2(C1)CN(C(C1CCC(=O)N1C)=O)C2 C(=O)(C(C)(F)CC)N(C1CCN(C(=O)CCNC(=O)NC)CC1)CCC c1(C(=O)OC)ccc(CC(N2CCCC2CN(C(=O)CN2CCCC2)C)=O)cc1 c1(C(=O)NC2C(CNC(CCCc3ccc(C)s3)=O)C2)ccccc1S(C)(=O)=O c1(C(=O)NCC2N(C(CCCCOC)=O)CCC2)cc2n(n1)CC(F)C2 N1(C(c2ccc(SC)o2)=O)C2CCC1C(NC(=O)CNC(c1ccccc1)=O)C2 c1(CNC(=O)NC2CCN(CCCOC)CC2)ccc2c(cnn2C2CC2)c1 C(=O)(CN=c1[nH]c2c(c(=NCCC3CCCO3)[nH]1)CCC2)NCCOC c1(C(C)C)ncsc1C(=O)NCC1(F)CC(NC(=O)C=CC2CCOC2)C1 c1(C(=O)NC2CN(CC(C3CC3)OCC)CC2(C)C)ccnc2[nH]cnc12 N1(C(C(C)CO)=O)CCCCC(C2CN(C(C3CCC(N(C)C)CC3)=O)C2)C1 CCCCCC(O)C(=O)N1CC2CCC1CN2C(=O)Cc1ccc(C)cc1 c1(N(C)CC2(CNC3CC(=O)N(C4CC4)C3)CC2)ccnc(CC2CC2)n1 C(=O)(CC(=O)N(C)CCOCCCNC(=O)CCc1nnc(C(F)F)o1)N(C)C N1(C(C2N(CC)CCC2)=O)CC(C2CC2)(C(N2CC(C)C(C)C2C)=O)C1 N1(C(C)C)N=C(C(=O)N2CCC3CN(C(C4(C)CC5CC5C4)=O)CC23)CCC1=O Cn1nc(CNC(=O)OC(C)(C)C)nc1C(F)(F)F.C1(CN(C)C(=O)O)CCC1 c1(C(=O)NCCNC(C(C(=O)OC)OC)=O)cc(Br)cc2scnc12 c1(C(=O)NCC(CNC(c2c(C)cc(C(F)F)o2)=O)(C)O)cccc(O)c1Cl CCC(C(=O)N1CC(O)(COC(C)=O)C1)NC(=O)CC1CNC(=O)O1 C1(NC(C(CCOCC)NC(c2coc(CC)n2)=O)=O)CC2CC3C(C2)C13 C1(C)(C(N2C3(CNC(c4c(C(C)C)cccc4)=O)CC(C2)C3)=O)CCN(C)C1=O c1(NC(=O)C(F)C2CC(NC(C3(F)CC=CCC3)=O)C2)cc(O)ccc1F C1(C(=O)NCCC(C)N(C(c2ncc(NC)nc2)=O)C)CCN(C)C(C)C1 S(=O)(=O)(c1cc(C#N)ccc1F)N1C2CN(C(C(C)O)=O)C(C2)C1 C(=O)(C(O)C(C)(C)C)NCC1(OC)CCN(C(c2ncc(C)cc2C)=O)C1 CCCC(CCC)CC(=O)NC1CCOC(CNC(c2cccn(C)c2=O)=O)C1 C1(C(=O)NCC2(C3CCC3)CC2)CCN(C(C2CC3OC2C2CC32)=O)C12CC2 N1(C(C=CCCC)=O)CCC(CNC(C2OCCC2(C)C)=O)C(CC)C1 c1(C(=O)NC(C(C(C)C)NC(=O)CCC2CCCCCC2)C)cccc(=S)n1O C#CC1(CNC(c2oc(CNC(=O)C(CN(C)C)CC)cc2C)=O)CCOCC1 N1(C(CCCC2CCCC(=O)N2)=O)CC2CC1CN2C(=O)Cn1nnc(=O)[nH]1 C1(CC(=O)NCCCN(C(CN(c2ccccc2)C)=O)C2CC2)CCS(=O)(=O)C1 N1(C(c2ccc(COC)cc2)=O)CCN(C(=O)CC2CC3CC3C2)CC1CO Cc1nc2ccc(OC(F)(F)F)cc2cc1C(N1C2CSCC1C2)=O N1(C(Cc2ccn(CC)n2)=O)CC(CNC(=O)CC=C(C)C)C(C)C1 n1(C(C)(C)C)ncc(C(c2nnnn2C2CCCC2)NC2(CCCCO)CC2)n1 C(=O)(CC(C)C(C)C)N1CCC(O)(CNC(c2c(C(C)=O)cnn2C)=O)C1 c1(C(N2CC(N(C(c3cc(C)cc(C)c3C)=O)C)C2)=O)cc(F)cc2ccoc12 c1(OC)ccc(C(C)=CC(=O)NCC(O)CNC(C2CN(CC(C)C)C2)=O)cc1 C(=O)(C1=NOCC1)NCC(C1CC1)NC(c1cc(-c2ccn(C)c2)[nH]n1)=O C(C)(CCC(=O)NCC1CCN1C(=O)Cn1cncc1C)SC C1(C(N2CCC(OC(F)(F)F)CC2)C(=O)NC2COC2)CC2CCC1C2 c1(C(c2nc(Br)c[nH]2)(C)C)ccc(F)cc1.c12cn(nn1)C1CN(C1)C2=O c1(C(=O)NCCC2CCN(C(CCSC)=O)C2)cc2c(o1)CCC(C)(C)C2=O C1(C(=O)NCC(CC)C#N)CC2(CCC2)CN1C(c1ccc(C#N)c(C)c1)=O CC(CC(N)=O)NC(=O)NCC(C1CCCCC1)F C#CCC(CC(=O)NCC1(c2ccon2)CC1)NC(C1CC(=O)NC(=O)C1)=O c1(C(=O)NC2CN(C(C(C(C)C)F)=O)CC23CC3)cc2ncn(C)c2cn1 Cc1cc([N+](=O)[O-])cnc1NC1CCCC(NC(c2c(F)ccnc2F)=O)C1 CCC(C)(CCC(C)C)C(=O)N1CC(CNC(c2ccc(CO)nc2)=O)C(O)C1 c1(CC(=O)NC(CCCNC(CCC(=C)C)=O)(C)C)c(C)[nH]c2ccccc12 n1(CC(=O)NC2CC3CCC2N3C(C2(F)CCOCC2)=O)nnc2c1CCCC2 N1(C(C(CC)N(CC)CC)=O)CCC(C)(NC(c2cnc(C(=O)O)cn2)=O)C1 CCC(C(=O)NCC(c1ccccc1)NC(=O)COC)C(C)(C)CC N1(C(C2C(OCC)CCC2)=O)CCCC(N=c2cc(C)nc(SC)[nH]2)C1 C#CC1(C(=O)NC(C)CC(C)NC(c2cscc2-c2ccccc2)=O)CCCC1 C1(CCC(=O)NC(C(=O)N(CC)COC(C)=O)C)Cc2ccccc2NC1=O.O c1(C(=O)NC(CNC(=O)CCc2ccoc2)C2CCC2)ncnc(O)c1Br c1(C(N2CCCCCCCCC2)C(=O)NCC)ccc([N+](=O)[O-])c(Cl)c1 C(C)(C)(CC(F)C(=O)N(C)C)NC(c1cn(-c2cc(C)c(=N)[nH]c2)nn1)=O N1(C(c2ccc(C(=O)OC)o2)=O)CCCC(N(C)C(c2ncsc2C)=O)C1 C1(NC(C(=O)NCc2ncn(CC)n2)=O)CCCCC1Oc1ccccc1 C1(N(C(C(C)OCC=C)=O)CC2CC3CCC2C3)CC2CCC(C1)N2 CN1CCc2cc(C(=O)NC(C3CCCN3C(=O)C=CBr)(C)C)ccc2C1 c1(OCCOC)ccc(Cl)cc1C(N1CC2CC(NC(C3CCCO3)=O)C1C2)=O C1(CC)CN(C(=O)C(C)Cn2cccn2)CCN1C(=O)CC1CCSCC1 CCCC(CCCO)C(=O)NC1CN(C(=O)CCn2c(C)csc2=O)CC1(C)C C(=O)(CCCCCCCS(C)(=O)=O)N(CCCCCNC(C(CC)C)=O)C CCCCS(=O)(=O)N1CCC(C(=O)NCC2CCN2C(C2CC(OC)C2)=O)CC1 Cc1ncc(Cl)cc1NC(C1(C(C)C)CCN(C(c2cnco2)=O)C1)=O c1(SCC)ccc(CC)c(O)c1.C12(CCCCC1)C(=O)N2.C12CCCC1C(=O)N2 c1(C(=O)NCc2cc(C(=O)NC3(CC#C)CC3)n[nH]2)ncc(C#N)cc1C C(C(C)(O)C(C)(C)C)NC(C(C1CN(C(Cc2n(C)ccc2)=O)C1)O)=O CC(C)CC(CNC(C12CCC(CC1)C2)=O)NC(C1CCN(S(C)(=O)=O)C1)=O Cc1c(C(=O)NC2CCCCC2NC(C2CCC(C)(C)C2)=O)cc(C2CC2)n1C CC(C)(C)CCCCNC(C1CN(C(C23CCC(OC)C2C3)=O)CC1(F)F)=O N1(C(CC(=O)NCC#C)=O)CCCC(N(C(=O)CC#N)CCO)C1 C1(CNC(C(C=C)OC)=O)CN(C(c2ccc(F)s2)=O)CC1(F)F c1(C(N2CCC(NC(c3[nH]cc(C)c3)=O)C2)=O)cnn2ccnc(N)c12 C1(C)(CNC(C2C(CC)OCC2)=O)CCN(C(=O)C(c2ccc(Cl)cc2)O)CC1 C1(C(=O)NCC2CCCC(CNC(c3nc(C)[nH]n3)=O)C2)C2CCC3C(C2)CC13 c1(C(N2C(C)CCC(NC(c3nc(COC)sc3)=O)C2)=O)nccc2ccsc12 C1(C(=O)NCCOCCNC(C2(C)CC=CCO2)=O)CC2(CCCCO2)C1 n1(CCOC)nnnc1C(c1cc(C2CC2)on1)NCCCCCC1CC1 c1(C(=O)NC2(CC=C)CCCN(C(=O)CNC(=O)NC)C2)ccc2nncn2c1 C(=O)(CS(=O)(=O)CCO)N1CC(C)N(C(c2[nH]c(=N)sc2-c2ccccc2)=O)CC1 C(=O)(C(C)(C)CC)N(C1CCN(C(=O)CS(N)(=O)=O)CC1)CC#C C1(CC)CC2CCC1O2.C1(C2CNC(=O)C3(COC3)C(=O)N2)CCCCC1 C1(NC(c2cc(F)cnc2O)=O)CC2CN(C(=O)CCn3cc(Cl)cn3)CC2C1 C1(COC)(NC(C2CC23CC3)=O)CCN(C(C2CCC(CC(F)(F)F)CC2)=O)C1 N1(C(C(C)NC(CC)(C)C)=O)CCCC1CN(C)C(C1(Br)CC1)=O C(c1ccncc1C)=CC(=O)NCC(CC)(C)NC(=O)CC(=O)N(C)C C1(NC(C(C)N(C)C)=O)CC2CC(C1)CN(C(c1cc(CF)on1)=O)C2 C(=O)(C(C)C(F)(F)F)N1C(C(CNC(c2c(CC)nc[nH]2)=O)(C)C)CCC1 C(=O)(C1=NOC2(CCC2)C1)NC1CC(NC(=O)CCN2CCCC2)C1 n1(CC(=O)NC2C(CNC(CNC(=O)OCC=C)=O)C2)nc(O)ccc1=O C1(OC)CCC(C(=O)NC(CNC(c2cc(CCO)on2)=O)C2CC2)C1 Cc1c(C(=O)NCC(F)CNC(=O)Cc2c[nH]nc2O)c(C(F)(F)Cl)nn1C C(=O)(CC(F)(F)C(F)(F)F)NCC1CCCN(C(C(CCCC)O)=O)CC1 CCCC(C(=O)N1CCC(CN(C)C(c2cnccn2)=O)C1)S(N)(=O)=O c1(C(=O)Nc2nnc(COCCOCC)s2)cccc(Br)c1 c1(C(=O)NC(C)CCCNC(=O)Cn2ncnn2)ccc2nnc(S)n2c1 c1(OC)c(CC(=O)N(C2CC3CCC(C2)N3C(=O)CC(C)C)C)cccc1C#N CCCC(CCC)CC(=O)NC1CC(CCNC(C2C3CCCC23)=O)C1 c1(C(=O)NC2C(C#N)CN(Cc3ccsc3)C2)ccc2ccc(Br)cc2n1 C1(C(=O)OC(C)(C)C)CCC2CN(C(=O)C(=O)Nc3cccc(CC(C)N)c3)CC12 O=C(CCc1cncs1)NCC1CC1CC(=O)NCC(F)CO C1(CC(=O)NC)CCN(C(=NC)NC2CC23CCc2ccccc23)CC1 c1(C(N2C(CNC(C3C(C#C)C3)=O)CC(OC)C2)=O)ccc2c(c1)CCOC2 C(C(C)(O)CC(=O)N1CCCC(N(C(=O)CCC(C)(C)F)C)C1)OC C1(=CCNC(c2csc(O)n2)=O)CCN(C(c2cccc(C(F)F)n2)=O)CC1 N1(C(C(C(C)C)OC)=O)CC(CNC(c2cnc(C(C)(C)C)o2)=O)OC(C)(C)C1 N1(C(Cc2cn(CC)nn2)=O)CC2CCC2(CNC(=O)C=C(C)C(C)C)C1 C1(CNC(C(CC#C)O)=O)CC2CCC(C1)N2C(=O)Cc1n[nH]c2c1CCCC2 c1(OC)cc(CN2CCCC(C(N3C(C)CCC3C)=O)CC2)ccc1OC C=CC1(CC(=O)NC2CCCN(C(=O)C(C)(C)C(C)C)C2)CCCCC1 CCCCCCCCN(C(=O)CCC1CC(NC(C2(C#N)CC2C)=O)C1)C Cc1c(Br)ccnc1C(=O)NC1CC1CNC(c1nsnc1O)=O C1(N(C(=O)Cn2cnc(C(N)=O)n2)C)CCCN(C(C2COCC2(C)C)=O)CC1 N1(C(CCNC(C(C)(C)C)=O)=O)CCC2CC1CN2C(=O)CC1CCOC1 CS(=O)(=O)c1cccnc1C(=O)NC1CCCC1NC(C1CC12CC(F)(F)C2)=O Nc1c(C(N2CCCN(C(=O)C=CC3CCOC3)CC2CO)=O)cc(F)cc1Cl c1(NC(=O)NC(C2(O)CCC2)C(=O)O)cnn(C(F)(F)F)c1 c1(N(C)CC2C(C)COC2)nccc(=NCc2ccccc2)[nH]1 C#CC1CCC(CNC(=O)NC2CC3CC(CO)CC23)CC1 Cc1cc(C(N2CCC2CNC(c2c(Br)noc2C2CC2)=O)=O)nn1C1CC1 N1(C(c2cccc(B(O)O)c2)=O)CCC(N2CCCC(O)CC2)C2(CC2)C1 N1(C(CC(C)c2cnn(C)c2)=O)CC2CCN(C(=O)C3=NOCC3)CCC2C1 C(=O)(C#CC(C)(C)O)N1CC(O)(CNC(C(C)SC(F)(F)F)=O)C1 c1(N2CCC(CC=C)(NC(=O)C(O)CSC)C2)cc(C)c(C#N)c(C)n1 CC(C)(C)C#CC(=O)NCCOCC(=O)NC(CO)CCO N1(c2c(C)cncn2)CCN(C(C23CC2COC3(C)C)=O)CC(O)C1 n1(CC(C(=O)NC2CN(C(CN(CC)CC)=O)C2)C)ncc2c1CCCC2 C1(NC(C(C)(C2CCC2)NC(CN2CC(C)(OC)C2)=O)=O)CCC([N+](=O)[O-])CC1 C1(NC(c2c(C)n(C)nn2)=O)C2CC3CN(C(=O)C4=COCCC4)C1C3C2 CC1(C)CC(CN)CN1C(=O)C(N1CCCC1Cc1ccccc1[N+](=O)[O-])=O C1(CC)CCN(C(c2ccnnc2C)=O)C1CNC(c1ncc(OC)cn1)=O C1(C(N2C(CCC(N3CCC(CF)CC3)=O)CCCC2)=O)CCCC12CCC2 C1(NC(C2C(c3nc(C)[nH]n3)C2(C)C)=O)CC2CN(C(=O)CC(C)(F)F)CC2C1 N1(C(CCCOCC)=O)CC(NC(c2cccc(C)c2Br)=O)CC(C)(C)C1 CCC(C(=O)Nc1cnn(CC2CC2)c1)NC(=O)C=CCF C(=O)(C1CCCc2[nH]cnc21)N1CCC(OCCNC(=O)CC(O)C2CC2)C1 C1(CC(=O)NC(C(=O)NCC=C)C2CC2)CCC(=O)NC1 CCCCCC(F)C(=O)NC(CC(N1CC(O)CC1(C)CO)=O)C1CC1 C(=O)(CC(C)COC(C)=O)N(C1CC(C(N(CCC)CCOC)=O)C1)C c1(CNC(C2C(C(=O)O)COC2)=O)c(Cl)ccc2c1OCO2 c1(C(N(C2CN(C(C(C)OCC=C)=O)CC2(C)C)C)=O)csc2c(O)ccnc12 C1(C)(CNC(C=CC(C)NC(c2cc[nH]n2)=O)=O)CC1(F)F N1(C(Cc2cc(C)sc2)=O)CCOC(C(N2CC(CO)C(C)(C)C2)=O)CC1 c1(OC)cnnc(C(=O)NCC2(NC(C3CCC(F)(F)C3)=O)CCCC2)c1 C1(C(N2CCC(NC(c3n(CC)ncc3Cl)=O)C(C)C2)=O)C2CCC3C(C2)CC13 c1(N(C(=O)CCC(N)=O)c2cn(C(C)(C)C)nc2)nc(-c2nn[nH]n2)c(Br)s1 CN1Cc2ccc(C(=O)N(C)CC3CCCCN3C(C3CC4CC4C3)=O)cc2C1 c1(C(=O)NCC(N(C(c2nccc(CC)c2)=O)C)C2CC2)cnccc1C#N c1(NC(=O)N(c2ccc(Cl)cc2)C2CCOC2)ccc(CCF)cc1 c1(COC)ncc(CN2CCCC=C(Cl)C2)c(C)n1 C1(CN(C)C(C2(n3cncn3)CC2)=O)CCCC(NC(c2cc(CO)on2)=O)C1 c1(C(=O)NCC(C)(C2CC2)NC(C(C=CC)O)=O)cc2c(C)ccc(F)c2[nH]1 C1(CNC(C(CC)COC)=O)CCCCN(C(c2ncoc2C)=O)CC1 n1(CCC=C)nc(C2CCC2)nc1-c1cncn1C C(=O)(C1c2c[nH]nc2CCC1C)NCc1cn(C2CN(C(C3C(C)C3)=O)C2)nn1 C1(NC(C2CC(CC)C2)=O)CN(C(=O)CCNC(=O)COC)CC2CCCC12 C1(CC)(NC(=O)COC2CCCCC2)CCCN(C(C2CCCC2)=O)C1 c1(C(N(C2CCN(C(C(CC)C)=O)CC2)CC(C)C)=O)ccc2cc[nH]c2n1 N1(CCNC(C2CSCCN2C(=O)CC2CCCC3CC23)=O)CCCNC1=O c1(CC(=O)N)c[nH]c2cnccc12.CC(=O)C(C)(c1ccccc1)c1ccccc1 CN=c1ccc(C(=O)NCC2CCCC2C(=O)Nc2cccc(OC)c2C)c[nH]1 C12(C(N3CC(CNC(=O)C4=CCC4)C3)=O)CC(CO)(C1)OC21CCC1 C1(N(C(C2CCCC2)=O)CC)CCN(C(=O)OC(C)(C)C)C1C1CC1 Cc1nc(Cc2ccccc2)sc1Cl N1(C(C2CC(OC)CN2C(=O)NC(C)(C)C)=O)CCCc2cc(Cl)cnc21 N#CC1CCN(C2CC2c2ccccc2)C1 Cc1c(Cl)ccc([N+](=O)[O-])c1NC(C12CC1CN(C(=O)CN1CCCC1)C2)=O CN1CC2CCCC(C1)N2C(C1CC(NC(=O)CC2(O)CCOCC2)C(O)C1)=O c1(C(=O)NC(CN(C)C(C2NC(=O)CC2C(F)(F)F)=O)(C)C)ncnc(O)c1Cl CC(C)CC(O)C(=O)NC(CNC(c1coc(C2CCCCC2)n1)=O)C1CC1 c1(C(C)C)cc(NC2CCC(NC(c3cc(Br)c[nH]3)=O)C2)ncn1 C1(F)(C(N(CC)CC)=O)CCCN(C(=O)CCc2ncccn2)C1 N1(C(c2cnn(CC)c2C)=O)CCC2CCC(C1)N2C(=O)CCCCCN=[N+]=[N-] N1(C(CCCNC(C)=O)=O)CC2CCC(CNC(=O)C(C)S(C)(=O)=O)(C2)C1 CCC(CC)C(F)C(=O)N(C(CNC(=O)CCC1CCCN1C)CC)C c1(C(N2CCN(C(=O)C(N3CCOCC3)O)C3(CC3)C2)=O)cccc2c[nH]nc12 Cc1nn(CC(=O)NCC(C)(O)CNC(C2CCCCO2)=O)c(=O)o1 n1(CC)cnc2c(N(CCS(N)(=O)=O)C)nc(N(C)CC3CCCS3(=O)=O)nc12 CC1CN2CCN1CC2C(=O)N(C(C)CCNC(=O)C(C)Cn1ccnc1)C C(=O)(CN=c1cc[nH]cc1)N1C(C(=O)NCc2cccc(F)c2)C2(C1)CCCC2 C(=O)(CC(F)(F)CC)NCC1(C(C)(C)C)CCN(C(C(=O)NCC)=O)C1 c1(CC)cc(C(=O)NC2CCC(C)(CNC(=O)CC3CS(=O)(=O)C3)C2)ncn1 C(=O)(CCCS(N)(=O)=O)NC1CCN(C(C2CCCN(C(CC)=O)C2)=O)CC1C C(CN=c1[nH]c(=NC)[nH]c(=NCC2(CC=C)CC2)[nH]1)SCCC=C Cc1ncc(C(=O)NC(C2CCCCC2)C(C)NC(=O)C(O)c2ccco2)s1 C(=O)(C(F)(F)C(C)O)NC1CC(NC(C2CC(C(=O)OC)C2)=O)CC1O C(N(C)N1CC(C(F)(F)F)CC1C)c1cn(COC)nn1 c1(CS(C)(=O)=O)cccc(C(=O)NCc2nc(C(=O)O)cs2)c1 c1(C(=O)NCC2C(NC(c3c(C)nc(C)s3)=O)CCCC2)cccc2[nH]ncc12 n1(CC)nc(C(=O)NCC23CC(CO2)N(C(=O)CN(C)C(C)=O)C3)ccc1=O C=CC(CC)CC(=O)N1CCC(CC)(NC(C2CC(CC)=NO2)=O)CC1 CCC(C)(COC)C(=O)NC1CCC(CNC(C2CCC(N(C)C)CC2)=O)CC1 C(=O)(N=S(C)(=O)C1CNC2(CCOCC2)C1)C1C(C)(C)C1(F)Cl Cc1c(NCC2CN(C(C)C)CCO2)ncnc1NCC1(Br)CC1 CC1CCOCC1C(N1CC(O)CC1C(=O)NCCc1ncccc1F)=O C(=O)(CC(CNC(c1coc(C(N)=O)c1)=O)C1CCC1)NCC(CC)OC C1(C(=O)OC(C(=O)NC(COCC)C)C)CCCCN1C(=O)OC(C)(C)C c1(NC(C2C3(CCN(C(c4n(C)ncc4)=O)C3)C2)=O)ccc2sncc2c1 Cc1cc(Cl)c(C(=O)NCC(CNC(C2CCC2C)=O)CO)cc1[N+](=O)[O-] C12(C(N(CC(C)NC(=O)CN3CC=CC3)C)=O)CC3CC(C(=O)N1)C2C3 C1(CC=C)(NC(C2CCCC2(F)F)=O)CCN(C(=O)CCc2c(C)noc2C)C1 c1(C(=O)NCC2CCC2NC(C2(CO)CCC2)=O)cccc2c1CCN2 C(c1cccc(OCC#N)c1)=CC(=O)NCC(CNC(C1(C)CC=CCO1)=O)F c1(C(N2CC(C)(NC(C3C4CCCOC34)=O)C2)=O)nn2cccnc2c1Br CN1C(=O)OCC1(C)C(=O)NNC(c1ccc(C(F)(F)F)c(C2CC2)c1)=O c1(C(N(c2c(C#N)cnc(C)n2)C2CCNC2)=O)c(C)nc2ncccn12 c1(Cc2ccnc(N(C3CCCCCC3)CC(F)F)n2)coc2cc(O)ccc12 C1(NC(c2cccc3nc[nH]c23)=O)CC2CN(C(c3ccco3)=O)CC2C1 N1(C(c2c(C)nco2)=O)CCN(CCNC(c2cnc[nH]2)=O)C2(CCC2)C1 c1(NC(=O)NCCCN2CCC(NC(=O)CC3CCNC3=O)C2)ccccc1Cl C1(C(=O)NCC(C(C)C)(C)NC(c2cnc(S)[nH]2)=O)CN2CCN1CC2 C1(CNC(COCCC=C)=O)CN(C(=O)Cc2ccc(Cl)cc2F)CCC1C N1(C(c2ccc(-c3ccc(C(=O)O)cc3)cc2F)=O)CCOC(C2CCCO2)C1 C1(c2ccc(OC)cc2)CCN(C(=O)CC(C)(F)F)CC1NC(C1CC(=O)N1)=O C(CC(C(=O)N(C)CC1CCCC2CC12)NC(=O)CSCC)=CC N1(C(c2ncc(F)cc2F)=O)CCC2C(C1)CN2C(c1ncn2c1COCC2)=O C1(CNC(CC2C(C)CC2)=O)CN(C(c2ccc(N)c(N)n2)=O)CC12CC2 c1(OC)cc(OC)c2c(c1)C(NC(=O)NC1CCc3c(C)nn(C)c3C1)CC2=O C1(NC(=O)CN(C(=O)CCCn2cncn2)C2CC2)CNC(=O)C12CC2 N1(C(c2c(C)snc2)=O)CCC2(CCOCC2)C(NC(C2CC3C=CC2C3)=O)C1 C(C)(C)(C(C)CC(=O)NC1CCOCC12CCC2)NC(CCC=C=C)=O C(=O)(C(C)CC(C)C)Nc1c(C(=O)OCC)c(-c2ccc(Cl)cc2)cs1 c1(-c2c(CCC)n[nH]c2)nc(-c2ccc(C)o2)nn1CCC N1(C(C(C)OCCC)=O)CC2COCC2(C(=O)Nc2ccc(C)nc2O)C1 C1(CCNC(=O)C2=CCCC2)CC2CCC(C1)N2C(=O)Cn1ccnn1 c1(N2CCN(C(=O)OCC)CC2)nc(Cl)nc(O)c1C C12CCCC1N(C)C2.CCCC(=O)NCC(=O)NCCSC(F)F N1(C(c2c(CC)ccs2)=O)CCCN(C(=O)Cc2csnc2C)CCC1 N1(C(=O)COc2cncc(Br)c2)CCN(C(=O)CCCF)C(C2CC2)C1 C1(C(N(C)CCOCCNC(c2ccsn2)=O)=O)C2Cc3ccccc3C12 N1(C(C2CC(F)(F)CS2)=O)CC2CC(NC(C3(CO)CCCO3)=O)C1C2 C1(N(C(=O)CC2CC=CCC2)CC#C)CCN(C(c2cnc(C)[nH]2)=O)CC1 C(=O)(CC(C(=O)NCC(C)N(C)C(c1cncnc1)=O)NC(C)=O)OC N1(C(C(C=C)OC)=O)CCC(C)(CNC(C23CC(F)(C2)C3)=O)CC1 C1(C(N2CC(C(N)=O)(CNC(Cn3ncc(C)c3)=O)C2)=O)CC(=O)N(C)C(=O)N1 c1(C(N(CCNC(c2c(CCC)nns2)=O)C2CC2)=O)cc(C)n(CCO)n1 c12ccc3nc(sc3c1)N(CCO)Cc1ccc-2cn1.Cc1[nH]nc(C(N)=O)c1C C1(CNC(C(CN(C)C)NC(CC=C=C)=O)=O)CCCN(C)C1=O c1(OC)cc(C=CC(=O)NC2CC23CC(NC(C2(F)CC=CC2)=O)C3)ccc1F C(CC(=O)N1CCC(NC(c2nc(C(C)C)oc2C)=O)C12CC2)(C(F)(F)F)OC CCC1=C(C(=O)NC2CN(C(c3cc(C(=O)OC)on3)=O)CCC2C)SCCO1 c1(CC(=O)N(CCNC(CNC(C(CC)CC)=O)=O)CC)cc(F)c(C)cc1F Cn1cc(C(N2CC(CNC(=O)Cc3ccsn3)C(C(F)(F)F)C2)=O)c(O)n1 N1(C(C2(CC(C)C)CCC2)=O)CC2(CCN(C(C3(C)COC3)=O)C2)C1 C1(C(N(C2COCC2O)C)=O)CN(C(C2CC(C)(C)CO2)=O)CC12CC2 N1(C(CC#N)=O)CCC2CN(C(c3ccc4c(O)n[nH]c4c3)=O)CC2C1 N1(C(C(C)OC2CC2)=O)CCCC1C(C)(C)NC(c1cc(C(C)(C)C)c[nH]1)=O C1(C(C)C)CN(C(C2CC(O)CN2C(N)=O)=O)CCC1NC(C1(CF)CCC1)=O N1(C(CCSCC(C)C)=O)CCN(C(C2CC(=O)N(CC3CC3)C2)=O)C2CCC12 C1(c2ccccc2)(C(N(C)CCNC(c2csc(CO)n2)=O)=O)CC(F)(F)C1 C1(C(=O)NCc2nc(CNC(c3[nH]ccc3C3CC3)=O)sc2)CN2CCC1C2 C1(Cl)(C(=O)NCC2(CNC(c3ccnc(S)c3)=O)CCC2)CC2CCC1O2 CC1CN(S(=O)(=O)c2ccc(NCCCC3CC3)c(Cl)c2)CC2(CCCCC2)O1 C1(NC(C2(CNC(C=C(CCN(C)C)Cl)=O)CC3(CC3)C2)=O)CCC(C2CC2)C1 C(=O)(CC(C(F)F)C(C)(C)C)N(C)CCNC(=O)C(C)(C)NS(C)(=O)=O c1(SCC(N2C(CNC(c3c(OC)cccn3)=O)CCC2)=O)nc(C)cc(C)n1 C(C1CCCCC1)=CC(=O)NC1C(CC(=O)N(C)Cc2nnnn2C)C(O)C1 CC1(C)CCN(C(C2CS(=O)C2)=O)CC1C(=O)NCCCc1ccsc1 C1(NC(CC2CC(N(C)C)C2)=O)CC(C(=O)NCC2CC23CC3(F)F)CC1O N1(C(C(CNC(C(CO)OC)=O)(C)C)=O)CC2CCC2(CO)C1 N1(C(C=C(CC)C)=O)CCN(C2(CN)CCOC2)CC1 N1(C(C)=O)CCC(n2cc(C(O)C3CC3)nn2)C(O)C1.O=C(CO)OC(=N)O c1(C(C(=O)NCC(CC=C)NC(=O)COc2cccnc2)O)ccc(F)c(F)c1 N1(C(C(C)SCC)=O)CC(NC(c2cccc(F)c2)=O)C(F)C1 N(C1CCCc2cc(NC(=O)OC(C)(C)C)ccc21)C(Cn1cc(C(C)=O)nn1)=O c1(CC(=O)N(C2CCCC(NC(c3c(C)ncs3)=O)C2)C)ccc2nonc2c1 N1(C(C(CC)(C)OC)=O)CCCCC12CN(C(=O)C(=O)C(C)(C)C)C2 C1(C)(NC(C2N(C(C3(C)N(C)CCC3)=O)C3C(C2)C3)=O)CC2CCC1C2 CC(C#N)CCC(=O)NCCCC1CCCCN1C(=O)CC1(O)CCCCCC1 C(CN=C(NCC1CC1)NC(C1CCCCO1)C)N1CCN(C(C)=O)CC1 C1(OCCC)CCCN(C(c2cc(CNC(=O)CCC(C)N(C)C)on2)=O)C1 c1(C(N2CC(C(C)NC(CCNC(COC)=O)=O)C2)=O)noc2c1CCCCC2 CCCCCCC(=O)N1CC2CC(NC(c3cc(=O)c(Br)c[nH]3)=O)C1C2 c12cccc(c1N(C)C)C1(CC)C(N(C(CC(C)(C)SC)=O)C)CN(C1)C2=O N1(Cc2cn(CC3(C(F)F)COC3)nn2)CC=CC12CCCC2 CC1(C(=O)NC2CC(C)(NC(C3CCCCO3)=O)C2)CCC(=O)C1 C(C1c2ccccc2CCN1C(c1c(C)nsc1C)=O)NC(C(CCSC)O)=O N1(CCCC)CCCC(C2CCN(C(=O)C(C(C)C)NC=O)CC2)CC1 CC1(C)CCc2cc(C(=O)NC(CNC(C3CC4C=CC3O4)=O)CO)ccc2O1 C1(CNC(Cc2ccc(C)s2)=O)CC(C(=O)NCC(C)C(F)F)=NO1 N1(C(CC2CC(=O)NC2)=O)CCC(NC(c2[nH]nnc2C2CC2)=O)C(O)C1 CC1(C)CC(N=c2ccnc(Cl)[nH]2)CN(C(=O)C(C)(C)N2CCCCC2)C1 C(=O)(C1=CC2(CCOCC2)C1)N(CCC)CCNC(=O)C(O)C(C)C C1(CCNC(CCSC)=O)CCCN1C(c1ccc(CN=[N+]=[N-])o1)=O.C(C=O)N Cn1ncc2c1CC(C(=O)NC1CCN(C(c3ccnnc3)=O)C1)CC2 c1(SC)cc(C)ccc1C(N1CC(CNC(=O)C(F)(F)CC2CC2)CCC1C)=O N1(C(CC2CN(C(C)=O)C2)=O)CC(C(N2CCCC2C2(C)CC2)=O)C(C(C)C)C1 Cc1nc(C(=O)NC2CC23CC(NC(c2c(C)noc2C)=O)C3)c2ccnc-2[nH]1 N1(C(C)=O)CCCC1(C)C(=O)NCC1CCCCN1C(C1(N(C)C)CCCC1)=O c1(C(=O)NCC(CNC(c2c(C)n(C)nc2Cl)=O)C)cccc2c[nH]nc12 Cn1cc(C(=O)NC2CCC(NC(c3cnc(C4CC4)nc3)=O)CC2)c(=N)[nH]1 CS(=O)(=O)c1nccc(N(C2CCCCNC2)C(=O)Cc2cncnc2)n1 c1(OCC)cc(C(N2CCC(CO)C(O)C2)C(=O)NCCC2CC2)ccc1OC CC(C)S(=O)(=O)CC(=O)NC(C)(C)CN(C)C(C1CC1Cc1ccccc1)=O C1(C(=O)NCC2(CC)CCOC2)CCCN1NC(=O)c1cncc(O)c1 C1(NC(C(Cn2cccn2)NC(COCC(=C)C)=O)=O)CN(C)CC1(C)C C(=O)(CCS(C)(=O)=O)NCc1cc(C(=O)NCC2(C)CCCC2O)n[nH]1 CC1=C(C(=O)NCC(C2CCCCC2)NC(=O)CCn2ccnc2)CCC1 N1(C(c2c(C)nc(COC)s2)=O)CC2CC(NC(=O)CCc3cnn(C)c3)C1C2 C(=O)(CCCCC(=O)OCCc1ccc(OC)cc1)OC.C12CN(C)C(=O)N1C2=O N1(C(C(C(=C)C)(C)C)=O)CC2CCCC2(Nc2ncnc(CC)c2F)C1 CC1(C)CNC(=O)C1NC(C1CCC(CNC(C2CCCC23CCC3)=O)O1)=O N1(C(C2C(C#N)C2)=O)Cc2occ(C(=O)NC3CC3C3CCCCC3)c2C1 c1(OC)cc(CNC(=O)C#CCNC(=O)CC(C)C2CC2)ncn1 c1(C(=O)NCc2scc(C(=O)NC(C(CC)C)C)c2)cc2occc2[nH]1 Cc1cc(C(N2CCOC(CC(=O)Nc3ccc(C(C)O)cc3)C2)=O)cc(C)n1 c1(CC(=O)NC2CCN(C(Cc3cc(C)sc3)=O)CC2)cccc2nonc12 c1(C(=O)NC2(CO)CN(C(c3c(O)cccc3F)=O)C2)cc(F)c(Br)cc1F Cc1cc(C(=O)NCC2CC3CC2CN3C(=O)C=CC2CCCN2C)nc(C)n1 c1(C(=O)NC2CC(CNC(C(C3CC3)OC)=O)C2)cnc2ccncc2c1 N1(C(C2(C(=O)NC)CCC2)=O)CC(N(C(=O)C#CC(=O)N(C)C)C)C(F)C1 c1(C(N)=O)nc(Br)cnc1NC(C1(C)CCN1Cc1ncco1)=O C1(C(=O)Nc2c(SC)cccc2)CC(C)CCN1C(C1CCCCC(=O)C1)=O c1(C(C)C(=O)NC2C3CN(C(c4ccncc4Cl)=O)CC23)c(F)cccc1F c1(C(N2CCC(O)(CNC(=O)CNc3ccccn3)C2)=O)ccc(O)c(CO)c1 C(=O)(C(C)C(O)CC(C)C)NCCCCC(=O)NCCNC(C(C)C)=O CCCC(C(=O)Nc1cccc(SC)c1)NC(c1cnc[nH]1)=O c1(C(N2CCC3(NC(Cc4scc(C)c4)=O)C(C2)C3)=O)c(S(C)(=O)=O)cnn1C Cc1nc(N(C)CCN(C(=O)C=CC(C)(C)C)C)cc(Cl)n1 c1(CN(C(=O)OC(C)(C)C)CCC2COC2)ccnc2[nH]ccc12 Cc1c(F)ccc(C(N2CCC(O)(C(C)NC(C3C4CC5C(C4)C35)=O)C2)=O)c1N C1(CNC(C2(NC(c3c(C)non3)=O)CCCC2C)=O)NC(=O)OC1(C)C C(=O)(C(CN(C)C)C(C)C)NCCCCC1CN(C(C(COC)OC)=O)C1 C(=O)(CC(CC(C)C)NC(=O)CC1CCCOCC1)N1C(CC)(CC)CCC1 c1(C(N2CCC(CCC(=O)N(CC(C)(F)F)C)C2)=O)cncc(O)c1 c1(CCNCC2(OC)CCCOC2)cccc2cc[nH]c12 c1(C(=O)NCC(COCC(=O)OC)(C)C)cccc(O)c1.C1(C)(C=O)CC=CCC1 CCCC(C(=O)NC(CNC(=O)CCN1CCCCC1=O)CCOC)S(N)(=O)=O N1(CCC)CC(C(N2CC3CC3(NC(C3CCC(=O)N3)=O)C2)=O)CC1=O C1(C)(CNC(C(C)CO)=O)CN(C(=O)CCc2nnc(C(F)F)o2)CCO1 C(=O)(C1CCCn2cnnc21)NC1C(CNC(c2ncc(C(C)(C)O)cn2)=O)CC1 N1(C(C(CC=C)CC)=O)CC(NC(=O)COc2cccc(O)c2)CC12CCCC2 N1(C(C(C)OC)=O)CCC(F)(F)C(CNC(=O)C(C)Oc2cccc(CO)c2)C1 c1(N(CCCOC)CCc2ccccc2OC)nnc(C(C)C)n1CC(C)C N1(C(C2OCCN(C(C)C)C2)=O)CCN(C(=O)C=CC2CC2)CC1CC(F)(F)F C1(C(=O)NC2CC(CNC(c3c(NC)snc3C)=O)C2)CCCCNC1=O c1(CC(=O)NCC(CC)NC(c2cnc(O)c(OC)c2)=O)c(F)cccc1Cl C(CCCS(C)=O)NC(CC=C)=O.C1C(=O)NCCS1 Cc1c(CCC(=O)NCC2(O)CC(CNC(C3C(Cl)(Cl)C34CC4)=O)C2)nnn1C c1(C(=O)NCC(C)NC(C2(CC#C)CCCO2)=O)cc(OC)cc[n+]1[O-] C12(CNC(C)=O)CCC(CN1C(c1ccc(C(C)=O)cc1F)=O)C2 N1(C(c2nc(CC)sc2)=O)CC2CC2(CNC(c2cnn(C)c2Cl)=O)C1 C1(=O)CS(=O)(=O)CO1.C1(C(C)C)CCCN(CCOC(C)(C)C)C1 C(CCCCCN(C)C(c1sc(Br)cc1F)=O)NC(C(F)=CCC)=O N#Cc1ccc(C(N2CCOCC2CNC(=O)Cc2ccsc2)=O)c(O)c1 CC(C)C(C(=O)NC1CN(C(C2CC(n3cnnc3)C2)=O)C1)n1cnnn1 c1(C(=O)NCCCC(C)NC(C(C(CC)O)C)=O)cncc2ccsc12 C1(F)(CNC(CC(C)c2ccccc2)=O)CCC(COCc2cccc(Cl)c2)C1 N1(C(C(=O)NCC)CCc2ccccc2F)CCC2CCC(O)C1C2 C1(NC(c2ccc(C(C)(F)F)cc2)c2n(C(C)C)nnn2)CC2(COCCO2)C1 c1(OC)cncnc1C(=O)N(C)CC1(O)CCN(C(=O)Cc2cc(C)nn2C)C1 N1(C(CC(C=C)C)=O)CCCC12CCN(C(c1ccc(N)c(F)c1Br)=O)C2 C1(C(=O)NCC2(O)CN(C(c3cnccn3)=O)C2)CC2(C1)CC21CC1 C1(CNC(c2c(OC)nsc2)=O)CN(C)CCN1C(c1cnn(C(C)C)c1N)=O c1(C(=O)NC2C(CNC(c3ncc(Cl)cc3Cl)=O)C2)ncn2c1CCCC2 c1(CCNC(CC2N(C(CN(C(C)=O)C)=O)CC2)=O)ccc(C)cc1 c1(C(=O)NCC2C=CC(NC(CC3C(C)C3)=O)C2)cc(C(F)F)n(C)n1 c1(N2CCN(CC(c3ccccc3)CO)CC2)ncnc2sccc12 C(c1cnc(O)nc1O)=CC(=O)NCC(C)N(C)C(c1ccc(Br)c(O)n1)=O N1(C(C(C)Oc2ccccc2Cl)=O)CCN(C(=O)CCn2cccn2)C(C)C1 n1(CC#C)c(C)cc(C(=O)NCC(C2CC2)NC(C2CCC(C)O2)=O)c1C c1(N(CCCN(C)C(c2cc[nH]n2)=O)C)ccc([N+](=O)[O-])cc1Br CC(CCC(=O)NOCc1ccccc1F)NC(C1CCN(C)C1)=O N1(C(c2scc(C)c2C)=O)CC2CCOC2(CNC(c2cc(N)ccn2)=O)C1 CC1CCN(C(c2ccc(CS(N)(=O)=O)cc2)=O)CC1CNC(=O)CSC(F)F C1(CNC(C2CC(=C)C2)=O)CN(c2nc(C)ncc2F)CCC12CCC2 CCC(C)C(C)C(=O)N(CCC(=O)NCc1ccc[n+]([O-])c1)C C1(C)(NC(N(CCCN(C)C)C)=O)CC(C)(C)C1 C1(C(N2CCC(N(C(=O)C(=Cc3cccs3)C)CCC)C2)=O)CCCC(F)(F)C1 C(=O)(CCCC(=O)NC(C)C)NCC(CNC(c1c(C)cc(F)s1)=O)O C(C)(C)(CC(=O)NC1CCOCC1C)N(C(Cc1c(CC)con1)=O)C N1(C(CCOC(C)C)=O)CCC(C)C(NC(C2CCS(=O)(=O)C2)=O)C1 C(C)(N=c1nc2c(cnn2C)c(NCc2sncc2Br)[nH]1)c1cnc(C)s1 N1(C(Cc2c(C)cc(Cl)nc2)=O)CCC(NC(=O)CC2=CCCC2)C(F)(F)CC1 N1(CCCNC(c2cnn(CC)n2)=O)CCN(C(=O)CC(O)C2CCCC2)CC1 N1(C(CC2CCC(C)C2)=O)CC2CC(NC(=O)C=Cc3cnn(C)c3)C2C1 C(=O)(C(=O)C(C)(C)C)NCC(CC(C)C)NC(CCCc1onc(CC)n1)=O CCC(CC)CN=c1[nH]c(=NC2CCCc3ccccc3C2)[nH]c2cc(OC)ccc12 N1(C(Cc2ccc(C)c(Cl)c2)=O)CCC(NC(C23CCC2C3)=O)C2(CCC2)C1 C1(NC(C(c2ccc(C)o2)C)=O)CN(C(c2ccnn2C2CC2)=O)CC12CCC2 c1(NC(C(CC)N(C)C(C2CC3CC3C2)=O)=O)ccc2nncn2c1 C12(CNC(=O)C3=CCCSC3)CN(C(=O)CC3CC3c3ccccc3)CC1CCO2 C1(CNC(C(COC)(C)O)=O)CC(C)CCN1C(=O)CN(c1ccnc(Cl)n1)C c1(NC(C(=O)N(C)CC2CCOC2)=O)ccc(C(=O)C(C)(C)C)cc1 C12(NC(c3c(F)ccc(C)n3)=O)CCN(C(C34CC5CC3C4C5)=O)CCC1C2 c1(NC(=O)CCNC(CO)CC(O)c2ccccc2)cc(F)cc(F)c1 c1(C(=O)OC)cc(C(N2C(C)C3CC2C3NC(C2CC2F)=O)=O)cc([N+](=O)[O-])c1 C12(C(=O)NC(CCC)C(=O)NC)CCCC1CCN2C(C1CC2(C1)CC2(F)F)=O CC(C)C(C(C)NC(=O)Cn1cnnn1)NC(=O)C=CCN1CCCC1 c1(C(N2C(C)CN(C(=O)COCC(C)(C)C)CC2)=O)cncc2n[nH]cc12 c1(C(N2CC=C(CNC(C3(C)CCC(C)C3)=O)CC2)=O)cc(F)c(N)c(F)c1 S(=O)(=O)(c1c[nH]ccc1=NC1CCC1C)NCCCNC(CC=C)(C)CC=C CC1=C(C(=O)N2CC(C)(C)CC2C(=O)NCC2(CO)CC23CCC3)CCC1 c1(C(=O)NCCCN(C(C(C)(C)C(F)F)=O)C2CC2)cc2c(s1)CCCC2 C1(C(=O)NCC2OCCN(C(C(C)(C)CC#N)=O)C2)CCCC2CCCN12 c1ccccc1F.C1(=O)C(=O)NCCN1.CCCCOCCOC(=O)CC C1(F)(C(=O)NCC2C(NC(c3cc(C(=O)OC)[nH]c3)=O)CCC2)C(C)(C)C1(C)C c1(C(N(CCC)CCNC(=O)CCCc2nccs2)=O)cc(C(N)=O)cc(F)c1 N1(C(C2(C)CCNC2=O)=O)C2CCC1(CNC(c1cnncc1O)=O)CC2 C1(NC(c2c(C)n(-c3ccc(F)cc3)nn2)=O)CCC(O)C(O)CC1 C(=O)(C1=NOC(C)(C)C1)NC(c1ccccc1)C=CCNC(CCCCCSC)=O c1(C(N2CC(C3(NC(C(CC)OCC)=O)CC3)C2)=O)ccc(F)c(S(N)(=O)=O)c1 CCC(CC)(C(C)C)NC(=O)C(C1CCCN(C(=O)C(O)CCSC)C1)C CCC(CC(=O)N1CCN(CC(C)NC(=O)C(C)=NOCC#N)CC1)CC(C)C C=CCC(C)C(=O)NCCC1CC(OC)CN1C(c1cncc(CO)c1)=O Cc1csc(=O)n1CCCC(N1CCCC(CNC(C2(F)CC2C)=O)C1)=O c1(OC)ccc(C(C)C(=O)NCC(C)(C)NC(c2cnco2)=O)c(C)c1 c1(C(=O)NC2C(C)CN(C(=O)Cc3cnnn3C)C2)cc2occc2n1C NC(CCNC(c1ccc(N)cn1)=O)CC(=O)N1CCOCC1 CC(C)C1=NOC(C)(C(=O)NCCC(C)N(C)C(c2ccnc(C3CC3)c2)=O)C1 CN1CCCC1C=CC(N1CCN(C(=O)C(=O)Nc2cccnc2)CC1)=O C(=O)(C(C)(O)C(F)(F)F)N1CC(CN(C(C(C)CCc2cccc(F)c2)=O)C)C1 c1(OCC)cc(C(N2CC(C)(NC(=O)COC(F)F)C2)=O)ccc1C c1(C(=O)NC(C2CCN(C(C(=O)NCC)=O)C2)C)c(F)ccnc1Cl c1(C(=O)OCC(C(=O)OC)(C)OC)cc(C)n(-c2cccc(F)c2)c1C N(C(=NCC1CCCC(OC)C1)N1CCC=C(c2ccco2)C1)C(COC)C c1(SCC(=O)NCC(C2CCCC2)NC(=O)CC2CC23CC3)nc[nH]n1 CC(C)C(C(C)NC(c1n[nH]cc1C1CC1)=O)NC(c1cnc(C#N)s1)=O c1(CC(N2CC(CC(C(=O)NC(CC)C)F)C2)=O)ncn(C)c1C C1(NC(CCc2n(C)cnn2)=O)C2CC1CN(C(=O)CCc1cnc[nH]1)C2 N1(C(C2CCC3(CC3)C2)C(=O)NC(CC)C)CCCCC12CCN(C)C2 n1(CC(=O)N(CCCN)Cc2ccccc2)ccc2ccccc12 C=CCC(C)C(C)(c1nnnn1CC=C)NCc1cccc(Cn2ccnc2)c1 C(=O)(CCC(=O)Nc1ncno1)NCC1CN(CC2C(C(=O)OC)CCO2)C1 c1(C(C(=O)NCCOCCN(C(=O)CN2CC(C)(C)C2)C)=O)cccn1C C1(CC)CN(C(C2CCC3(CC3)C2)=O)CCN1C(=O)Cn1ccc(C(F)(F)F)n1 N1(C(c2csc(-c3ccco3)n2)C(=O)NCC)CCc2ccc(Cl)cc21 Cc1nsc(C)c1C(=O)NCC(F)CNC(c1cccc(-c2cscn2)c1)=O CC1CN(C(=O)C(C)(C2CC2)N(C)C(C2CNC(=O)O2)=O)CCN(C)C1 C1(CNC(N2CCC(c3ccc(C)cc3)CC2)=O)COc2ccc(F)cc2C1 N1(C(CC2CN(C(c3c(C)nco3)=O)C(C)C2)=O)CCOC(C)C1C N1(C(C(C)C2CCC2)=O)CC2(C(=O)Nc3cc(Cl)cnc3O)CC1CCO2 CC1CC(C(N2CCC2C(=O)NC(C)CC2CC2)=O)CC(=O)N1 Cc1ncc(C(N2CCC(NC(c3nc[nH]c3C(F)(F)F)=O)C2)=O)c(C(C)C)n1 N1(C(C(c2ccncc2)C)=O)CCC2(NC(c3cc(Cl)ccn3)=O)CCCC12 c1(-c2nccc(C(=O)NCC(c3cccc(O)c3)O)c2)ccc([N+](=O)[O-])nc1 c1(COC)cn2c(n1)CCC2.N1(C(C2CC3N2C3=O)=O)CC2CCC(C1)O2 n1(CC)nc(NC(=O)N(C2CCN(Cc3ccccc3)C2)C)cc1C1CC1 N1(C(C(COC)(C)O)=O)CC(C(C)C)CC(CNC(=O)C(C)(C)n2cccn2)C1 C(C(F)CNC(=O)C(C)SC)NC(COCCOCCOC)=O.c1ccco1 c1(C(N2CCC(C(C)(C)NC(=O)C=Cc3cscn3)C2)=O)cc[nH]c2nccc1-2 N1(C(CSCC=C)=O)CCC2(CCCC2CNC(=O)C(F)CC)CC1 N1(CC)C(=O)CCC1CC(=O)NCC(C)NC(=O)COCC(F)F C12(NC(c3c(CC)non3)=O)CCCC1N(C(c1ccc(O)c(OC)c1)=O)CC2 N1(C(c2cn(CCNC(C3(Cl)C(C(C)=O)C3)=O)nn2)=O)CCC(O)C(F)C1 C1(CNC(c2cccc(N)c2)=O)CCN(C(=O)C=Cc2ccncn2)CC1O CCCCCCCCC(=O)N1CCCC(CN(C)C(c2ccc(N)c(F)c2)=O)C1 N1(C(=O)OC)CCCC1C(=O)NCC1(O)CN(C(C2C(C)C2C)=O)C1 c1(-n2c(-c3cc(C4N(C)CCC4)on3)nc(CC(C)(C)C)n2)ccc(C#N)cc1 c1(C(=O)OCC(C2C(C)(SC)C2)=O)cc2c([nH]1)CCOC2 C1(C(N2CCC(NC(c3c(C)nc(C(C)C)s3)=O)C2)=O)CCC(C2CCC2)CC1 FC1(F)CC1C1CCCN(C(=NCCCCl)NCc2cccc(C(F)(F)F)c2)C1 C1(CC)CN(C(=O)C(=O)NC(C)C)CCN1C(=O)CC1COCCO1 C(=O)(C(C)C(=O)N1CC2(NC(=O)CCc3ccc(F)nc3)CC1C2)OC c1(NCC)ccc(CNC(N2C(C)CCC2C)=O)cc1 C1(C)(CCNC(C=CC=C)=O)CCN(C(=O)CCOC(C)=O)C1.C(C(C)C)O N1(C(C(c2n(C)cnc2)O)=O)CC2CC(NC(=O)CNS(N)(=O)=O)C(C2)C1 N1(C(C(C)N(C)C)=O)CC(O)(CCNC(=O)C(C)C2CCCC2)C1 CC(C(=O)N1CCCc2ccnn21)N(C)C(C1C2CC3C(C2=O)C13)=O c1(OC)ccc([N+](=O)[O-])cc1C(=O)NCC(C)(CO)NC(=O)C(C)CC(N)=O Cn1cnc2c1CCCC2C(=O)NC1CS(=O)(=O)C1(C)C c1(CNC(=O)NCC(C)F)cc2sc(Cl)cc2[nH]1 c1(CC(=O)NCC(CNC(c2c(CC)cnn2C)=O)(C)C)c(C)cccc1Cl c1(C(=O)NC2C3(CC(NC(C=C4CCC(C)C4)=O)C3)C2)ccc2[nH]c(=N)[nH]c2c1 c1(C(=O)NCC2N(C(C(C)OC)=O)CCCC2C)oc2ccccc2c1CO C1(C(=O)NCCC2(NC(C(C)SC(C)C)=O)CC2)COCCN1NCC1CCC1 N1(C(c2c(C)ccc(C(F)F)c2)=O)CCC2(CC(NC(=O)C#CC(C)C)CO2)C1 N1(C(CS(C)(=O)=O)=O)CC(C2CCCCN(C(c3cnc[nH]3)=O)C2)C1 C(=O)(C1=CC2(CCN(C(=O)CNC(N)=O)C2)C1)NC(CC=CC)CO CN=c1[nH]cc(C(=O)NC2CC=CCC2C(=O)Nc2cnn(C)c2C(C)C)o1 C1(NC(C(C)(C)SC)=O)CCCC(NC(=O)COCC(C)(C)C)CC1 C1(C(=O)NC(C2CCCC2)CNC(C2(CC)CCC2)=O)COCC(C)O1 N1(C(C(CC)C(C)C)=O)CC2CCN(C(=O)Cc3ccc(OC)cc3F)C2C1 C1(NC(CN(CC)CC)=O)CN(C(C2CC(C)CCO2)=O)C2(CCOCC2)C1 C1(NC(c2c(C)cncc2)=O)CCC12CN(C(=O)Cc1ccc(F)c(Br)c1)C2 N1(C(C(C)(C(=O)OC(C)(C)C)OC)=O)CC2CN(C(=O)C(C)=C3CC3)CC2(C)C1 N1(C(C(C)SCC)=O)C(C(=O)Nc2ccc(F)cc2)CCC12CC2 C(C(C)(C)CC(=O)N(C(CC(C)C)C(=O)N(CC(F)(F)Cl)C)C)OC c1(C(N(C(CNC(CCc2ncc(C)[nH]2)=O)C)C)=O)cccnc1O c1(C(=O)NC(CC(C)NC(C2(OC)CCOC2)=O)C)cc2cc(Cl)ncc2[nH]1 c1(C(N2CCC3C(C(N4CCCC4C(F)(F)F)=O)C3C2)=O)cnc2ccccn12 CC1CN(C(=O)CCN(C(=O)C(C)c2cccs2)CC2CC2)C(C)C(C)(C)O1 C1(C2CC2)(CNC(C=Cc2cn(C)nn2)=O)CCN(C(C2CCSC2)=O)C1 c1(CC)[nH]ccc1C(N1CC(=C(F)CNC(=O)C(C)C2CCCC2)C1)=O C1(CNc2ncc(-c3ccc(CNC(C)=O)s3)cn2)CCC(C)=C(C)C1 N1(c2ncc(C(=O)OC)nc2)CCCC(C)(C(=O)NCc2ccc(Cl)c(Cl)c2)C1 N1(C(c2cnc(C)o2)=O)CC2CCC(N(C(=O)C=Cc3ccc(C)o3)C)C2C1 n1(C(C=C)C)nc(Cc2ccc(OC)cc2)nc1C1(c2ccc(Cl)cc2)CCC1 c1(CCn2cc(SCc3nccc(C(=O)OC)c3F)nn2)cnc2ccccn12 c1(CC(=O)NCC(C2CCCC2)NC(C(C)=C2CC2)=O)nc(C2CC2)n[nH]1 c1(C(c2n(C3(C)CC3)nnn2)NCC(C(C)C)c2cccnc2)cccc(F)c1 N1(C(C=Cc2ccc(C)o2)=O)CCC2(NC(c3nccs3)=O)CCCCCC12 N1(C(CCCN(C(=O)CCOC2CCCC2)C)=O)CC2(CCOCC2)C1 C1(CC(=O)NC(C(C)NC(CC2(COC)CC2)=O)(C)C)C(=O)NN=C1C N1(C(c2n(CC)nnc2)=O)C2CCC1C(F)C(NC(=O)C(CC)(CC)OC)C2 C1(C(N2CCC(N(C(C(C)=C(CC)C)=O)C(C)(C)C)C2)=O)CCC(C)(C)O1 C(=O)(CCCC(C)=O)N1C2CC(NC(C=COCC)=O)(C2)C1 n1(CCC(=O)NC2CCN(C(=O)CC3(O)CC3)CC2CO)ccc2ccccc12 c1(C(N(CCCN(C(=O)C(F)C(F)(F)F)C)C)=O)ccc2c(c1)C(C)(C)CN2 c1(NC)ccc(Cl)c(C(=O)N(CCCNC(=O)CC2CC3CCC2C3)C2CC2)c1 CN1CCC(C(N2CC=CC2C(=O)NC2CC(O)(CO)C2)=O)CC1=O C=CCCCCCC(=O)N1CC(O)(CN(C(=O)CSc2ccc(O)cc2)C)C1 c1(CC(N2CCC(CNC(c3ccc(COC)[nH]3)=O)C2)=O)ccc(F)c(Cl)c1F N1(C(Cc2ncc(CC)[nH]2)=O)CC(NC(c2cc(C)nn2C2CC2)=O)CCC1C C1(NC(C(C)SCC)=O)CC(=O)N(C2CN(C(c3cocc3C)=O)C2)C1 N1(C(Cc2c(C)ncs2)=O)CC(NC(=O)CCc2cccnc2F)CC1(C)C c1(C(C=CC(=O)NC(CC)CNC(c2cc(OCC)cs2)=O)=O)ccc(N)cc1 Cc1nc(C(C)C)cc(=NCC=CCNC(c2ccccc2C(=O)N(C)C)=O)[nH]1 c1(C(N2CC(NC(C3C(SC)CCC3)=O)(CO)C2)=O)ncn(C)c1C C1(C(C)NC(=O)COCCF)CN(C(c2cc(-c3cnccn3)[nH]n2)=O)CCO1 C#CC1CCC(C(=O)N(C)CCN(C(=O)CCC2CCCO2)C)CC1 c1(CC(C)C(=O)NCC2CCN2C(=O)CCNC(=O)C=CCl)cccc(F)c1 C1(C(N2CCC(CC(=O)N(c3ccccc3)CCO)C2)=O)Cc2c[nH]cc2S1(=O)=O C(=O)(C(C(C)(C)C)NC(=O)COC1CC1)NC(C(C)C)CO C1(C(=O)NCCCN=[N+]=[N-])CCCCCN1C(=O)CCc1ccccc1 C1(NC(c2c(C)cccc2)=O)CC2C1CCN2C(c1ccc(C)c(O)n1)=O c1(CCC(=O)NCC(C2CC2)NC(C2C(Cl)(Cl)C23CC3)=O)ccc(O)c(Cl)c1 C1(Cc2nnc(C)o2)CCCCC1C.C12CCCN1C(=O)CN(C)C2(C)C Cc1cc(NC(c2cc(C(=O)N(C)C)c(N)cc2F)=O)c(C)c(Cl)c1C C1(C(=O)NC(CC)CO)CN(C(c2nnccc2C)=O)CCN1C N1(C(CCc2cnc(C)s2)=O)CCN(C(c2csc(Cl)c2)=O)CC1CF c1(C(=O)NC2(C)CC(NC(CCCCN(C)C)=O)C2)n[nH]c2c1CCOC2 c1(NC(C(C)C)CCN(C(=O)Cc2ccccc2)C)nc(C(C)C)ccc1C#N c12ccc(cc1)c(=O)[nH]2.c1(CC(=O)NCCC(N)=O)ccccc1N c1(C(=O)OC)[nH]nc(-c2ccc(Cl)s2)c1-c1nn[nH]n1 N1(C(C2CCCN(C(C3CC(C(=O)NCC)C3)=O)C2)=O)CCC(OC)C(C)C1 C(CN1C(=O)Cc2ccccc21)NC(C1CCCCC(F)(F)C1)=O Cc1nc(C)n(CCCC(=O)NC(C)CC2CN(C(=O)C3=NOCC3)C2)n1 n1(C(C)C)cnc2c(N(CCF)C3CC3)[nH]c(=NCC3(C)CC4CCC3C4)nc12 c1(C(C(=O)NCCOCCNC(C(C)OCC=C)=O)(C)C)ccc(C)cc1 Cc1ccc(F)cc1-n1cc(CCNC(c2cc(F)cc(Cl)c2)=O)nn1 c1(Nc2ncc(CCNC(c3ncccc3Cl)=O)s2)ncncc1I CC1=C(C(=O)NCC(C)NC(=O)C(C)Oc2ccc(C)cc2)SCCO1 CC1CN(C(=O)C(=O)NC2CC2)CC1NC(C1CC1(C)Br)=O c1(C(=O)NCC2C(NC(=O)C=Cc3ccccn3)CCCC2)cc(F)cc(Cl)c1 CC1C(NC(c2cc3c[nH]cnc-3n2)=O)CC2CCC1N2C(=O)Cn1cccn1 N1(C(c2ccc(C(C)C)cc2)=O)C2CCC1C(F)C(NC(=O)CN=S(C)(C)=O)C2 c1(C(=O)NCC2N(C(c3ccc(=N)[nH]c3)=O)CCC2)cn(CCO)c(=O)nc1O N1(C(CCC=CC)=O)CC(NC(C2(C)CC2(F)F)=O)C(C(F)F)C1 C1(C(=O)NCCN2CC=C(C)CC2)(NCCOC)CCN(C(=O)C2=C(C)CCC2)CC1 C1(C(=O)NC(C)CCN(C(=O)CCSC(F)(F)F)C)CCc2ccccc2C1 CC1CN(C(C2(C)CCCS2)=O)CC(C)N1C(=O)Cc1nc[nH]n1 c1(-c2cc(C(=O)OC)c(CO)cc2)ccc2nc(N3CC(C#N)C3)sc2c1 CC1CCN(C(=O)CCC2CCCN2C)CC1NC(=O)CS(=O)(=O)NC1CC1 N1(C(=O)NCc2cc(C)c(Br)nc2)CCCNC(=O)C1C N1(C(CC2C(=O)NC(=O)N2)=O)Cc2occ(C(=O)NC3CC4(CCC4)C3)c2C1 CCCCCCCCCC(=O)N1CCC(CNC(=O)CCC2CC(OC)C2)CC1 N1(C(C(C)N(CC)CC)=O)C2CCC1CC(O)(NC(=O)C(C(C)(C)C)N(C)C)C2 C1(NC(C(CCC)C(=O)OC)=O)CCN(C(C2(C)CC2(F)F)=O)CC12CCC2 Cc1cc(C(=O)N(CCCN(C(=O)COCc2ncc(C)o2)C)C)cnn1 C1(C(C)C)N(C(c2ccncc2N)=O)CC12CCN(C(=O)C(C)(Cl)Cl)CC2 N1(C(COCCC=C)=O)CCN(C(=O)CN2CCC(O)CC2)C2CS(=O)(=O)CC12 C1(CN(C(=O)C=Cc2ccco2)C2CC2)CC2CN(C(=O)CC3CCCO3)CC12 n1(C(C)C(=O)NCCC2CN(C(C3COCCN3C)=O)C2)cc2c(n1)CCCC2 Cn1cc([N+](=O)[O-])c(N2CC3CC(NC(c4cc(Cl)c[nH]4)=O)CC3C2)n1 N1(C(=O)NC2CCN(C(=O)OC)CC2)CC2CCN(c3ncc(Br)cn3)CC2C1 C(CC(=C)C)(C(=O)OC)NC(C1(CNC(C(C=C)O)=O)CCCC1)=O c1(C(N2CCN(C(c3cc(CCC)[nH]n3)=O)CC2C)=O)cc2ccc(Cl)cc2[nH]1 c1(C(=O)NC2CN(C(c3ncc(CC)nc3)=O)CC3C2C3)cn2nc(C)sc2n1 N(C1CCCc2ccoc21)C(C(C1(O)CCC1)NC(CC(C)c1ccco1)=O)=O C(C)(C(=O)N(C)CCN(C)C(C1(c2cc[nH]n2)CC1)=O)OCCCC N(C(=NCCCCC(F)(F)F)NCC1CC2C(C1)C2(F)F)C1CCN(CC)C1 O=C1CC(C(=O)NC2CCCCN(C(=O)C(F)CC3CC3)C2)NC(=O)N1 C(=O)(C1=C(C)OCC1)NC1CC(CC(N2CC(C(CC)CC)C2)=O)C1(C)C C12(NC(C3C(C#N)CC3)=O)CC3CC(C1)CC(NC(C1CC(O)C(F)C1)=O)(C3)C2 CCC(O)CC(=O)NCCCC(C)NC(c1ccc(-c2nc(C)no2)cc1)=O C1(C(=O)NC(C=C)C)CC(O)CCN1Cc1ccc(N2CCOCC2)s1 c1(CNC(C2C(C)(C)C2)=O)ccc2c(c1)CCN(C(=O)C=CCN1CCC1)C2 n1(CC)ncc(Br)c1C(N1CC(N(C(=O)C2=CCCS2)C)C(F)C1)=O C1(NC(=O)OC(C)(C)C)CC(C(=O)OCC(c2ccc(Br)cc2)=O)=NO1 CC(O)C(C(=O)NC1COCC1C(=O)NC(C1CCCOC1)(C)C)N(C)C C(CCC)(CCCNC(c1ccc(CO)cn1)=O)NC(c1c(CCC)n[nH]c1)=O C1(C(=O)NC2C3CN(C(C4(NC(C)=O)CCCC4)=O)CC32)CCCCC1(C)C N1(C(c2c(COC)cc[nH]2)=O)CCC2C(C1)CN2C(C1CN(C2CCOC2)C1)=O N1(C(CC(=C=C)C)=O)CCN(C(c2ccc(Br)o2)=O)C(c2ccccn2)C1 Cc1cc(NCC2CC2)ncc1NCCN1CCOCC1 N1(Cc2c(CNC(=O)OC(C)(C)C)ocn2)CCc2cc(Cl)ccc2C1 Cn1cc(CC(=O)NC(C(=O)NCC2SCCS2)c2ccoc2)cn1 N(C1CCSc2ccc(Br)cc21)(C(=O)CC1CS(=O)(=O)CCN1)CC CCC(CNC(c1ccc(N)cn1)=O)(CC)NC(=O)C(CC1CC1)OC C(N=c1[nH]c2c(c(=NC(C)CSC)[nH]1)CCCCCC2)C1(OC)CCCOC1 N1(C(C(CNC(=O)OC(C)(C)C)C(F)(F)F)=O)CCN(C2CC2)CC(C)(C)C1 N#CC1CN(C(=O)Cc2cc(-c3nccs3)ccn2)CCO1 c1(OC)ncc(CN2CCC2C(=O)NCC2CCCOC2)cc1Cl CC(C)(C#N)CC(=O)N1CCC(CC(=O)NC2(C(C)(F)F)CC2)CC1 N1(C(CSCCOC)=O)CCC(F)(CNC(=O)CC2CCC(C)(C)CO2)CC1 c1(C(c2nnnn2CC(F)F)N(CCCO)CC2CCC2)ccc(Cl)c(Br)c1 CC1CN(C(=O)C(C)C(F)(F)F)CCCN1C(c1c[nH]c(C(N)=O)c1)=O c1(C(=O)NC2C3N(C(C45CC(C)C4C5)=O)C(CC3)C2)ccc2c(c1)ncn2C Cc1sccc1N(C(c1ccc(C2CC2C)o1)=O)C(C)C c1(CNC(=NC)NCc2ccc(-n3ccnc3)cc2C)ccc2ccccc2c1 c1(OC)ccccc1SCC(=O)N(CCCNC(=O)CC1COC(=O)N1)CCO C(C)(C(=O)NCCO)OCC(C)O.C1C(=O)NCCN1CC CC1(C)CC(C(=O)NC2CCCC2NC(c2cc(C(F)F)cs2)=O)CC(C)(C)O1 CCC(C)C(=O)C(=O)NOCC(=O)N=c1ccn(CC(C)C)[nH]1 C(=O)(C1=C(Cl)CCOC1)N1CC(N(C(c2cnc(C)n2-c2ccccc2)=O)C)C1 C1(CNC(COCC)=O)CC2(CCC2)CN1C(=O)C(CC)(CC)c1ccccc1 C(C=CC(=O)NCCN(C(=O)C=CCOC)CCOC)(CC)=CC N1(C(C(=O)NCCCCCC)C(C)CC2CCCC2)CCN(C)C2(CCOC2)C1 CCCC(C(=O)N(C1CC(C)(C)C1)C)NC(C1CC1(Cl)Cl)=O C(=O)(C(CC)CC)NCC1CC(F)(CNC(C(F)=CC)=O)C1 C(=O)(CC(C)(C)C(=O)OC)N1CC(C(N(C(C#C)C)C)=O)C(C)(C)C1 N1(C(C(c2cn(C)nn2)NC(C(CCC(C)C)=O)=O)=O)CCc2c(nnn2C)C1 CCC(C(=O)NC(C)CN(C(c1nncn1CC)=O)CC)C(C)C C1(C(N(CCNC(c2ccc(CC)s2)=O)CC)=O)CC2(CCO2)C1 c1(-c2ccc(C#N)cc2)cc(C(=O)Nc2cnc[nH]2)c2cn[nH]c2c1 N1(C(CC)=O)CCOCC(F)(CNC(c2ccc(-n3cncn3)c(N)c2)=O)C1 c1(NC(C(c2ccccc2)NC(CNC=O)=O)=O)ccc2c(c1)CCO2 c1(C(C)N(CCN)CCN)ccc(Br)cc1 c1(C(=O)NCCOCCOCCCNC(CC(=C)C)=O)ccc(C)c(CO)c1 N1(C(c2c(CC)cno2)=O)CCC(F)(CNC(=O)CCC2CCC(=O)N2)C1 N1(C(CC2(C)CC2(F)F)=O)CCCC(CCNC(=O)Cc2ccc(O)cc2)C1 C(C)(C(=O)N=c1cc[nH]cc1N1CCN(C)CC1)OCC(C#C)C Cc1cc(Cl)ccc1CC(=O)NCC1COCCN(C(=O)COCCF)C1 c1(C(N2CC3C(NC(c4c(Cl)n[nH]c4C4CC4)=O)C3C2)=O)cc(Cl)c(F)cc1O C1(CCNC(=O)CN2CCOC2=O)CCCCN1C(c1cc(Cl)n[nH]1)=O C1(NC(C2(CC=C)CC2)=O)COCC1C(=O)NCCCC1CCOC1=O C=CCCCC(=O)N(CCN1CCN(C(=O)CC2CC2C(F)(F)F)CC1)CC C(=O)(C(F)C(C)C(C)(C)C)N1CCC2(CN(C(c3ccc(CC)s3)=O)C2)C1 C(=O)(CCCSC)N(C(C)CNC(c1c[nH]nc1-n1cnnn1)=O)CC c1(CN2CCC(C(N3CCCN(C(=O)OC)CC3)=O)CC2)cc(Cl)c(Br)cc1Cl N1(C(c2c(CC)cc(N)cc2)=O)CC2CC(NC(=O)CCC(C)O)CC1C2 c1(C(N2CCCC(N(C(c3ccc(OC)cc3)=O)C)C2)=O)cc(Cl)ccc1O C(c1ccc(Cl)cc1Cl)=CC(=O)NCC1CCN(C(CN(C)C(N)=O)=O)C1 C(=O)(C1=NOC2COCC12)N1C(C)CC1C(=O)N(CC(C)(C)C#N)C Cc1cncnc1.c1(CC(=O)N2CCCNC2=O)n[nH]c(C)n1.C1CC1 c1(OC)cc(C(N2CCC(C(N3CCCOC(C)C3)=O)C2)=O)cc(OC)c1Br C1(C(N2CC(CNC(CC3CC(C)(C)OC3)=O)OCC2)=O)CCCC(F)(F)C1 c1(CC(N2C(CO)CC(NC(CCC(C)(F)F)=O)C2)=O)coc2cc(Cl)ccc12 C1(OC)CN(C(C2(C)CC(N(C)C(=O)OC(C)(C)C)C2)=O)CC12CCOCC2 N1C2CCc3cc(ccc3CC2)NC1=O.c1(C(=O)OCC)snc(OC)c1Br N#Cc1cc(C(=O)OCC(=O)N(CCC#N)CCC#N)cs1 c1(OCCC)ccc(C(=O)N(CC(C)NC(=O)C#CC2CC2)CC)cn1 c1(N(CCCCN(C(C2(COC)CC2(F)F)=O)C)C)ncn(C)c(=O)c1Br c1(CC(N2CC3C(CNC(=O)COCCF)C3C2)=O)cnc2cccnn12 Cc1cc(C(=O)NC2CC(C)CN(C(=O)CC3CCS(=O)(=O)CC3)C2)cnc1C c1(-c2onc(CCCF)n2)cc2n(n1)CC(O)CO2 c1(CC(=O)N(CCC(=O)O)C(C)C)sncc1Br c1(C(=O)NC(C2CCCO2)CC)n[nH]c2c1CN(C(=O)CN1CCC(F)CC1)C2 c1(C(N2C(C(C)C)CN(C(C3CC4CC4C3)=O)CC2)=O)cc(=O)n2ccsc2n1 Nc1c(C(=O)NCCC(O)CNC(=O)CC2CC2(Cl)Cl)cnn1CCO C1(OC)(CNC(=O)C(C)(C)c2cnc[nH]2)CCN(C(c2ccc(=N)[nH]n2)=O)C1 C1(C(N(CC(C)C)CC(=O)NC2CCC(O)CC2)=O)CC(=O)CC12CCC2 N1(C(C(C(C)O)(F)F)=O)CC2CCCC2(CNC(c2cn(C)c(=O)n2C)=O)C1 CC1CCN(C(=O)CC(C)(O)C2CC2)C(C)C1NC(C1CCCC2CCCN12)=O c1nn(C2CC2)cc1C(c1nnnn1C1COC1)NC1CC2CC2C1 C1(C(=O)NC(C(C)NC(c2c(OCC)cccc2)=O)C)CCCN2CCCC12 CCCCCC(C(=O)NCC1CC1CNC(=O)C=C1CN2CCC1CC2)C(C)C c1(CNC(c2c(SC)ccs2)c2nnnn2C)ccc(CC#N)cc1 c1(CC)cnoc1C(=O)NCCN(C(c1cc(COC)on1)=O)CC1CC1 c1(C(N2CCN(C(=O)C(C3CCC(=O)N3)C)CC2)=O)cccnc1OC(C)C C12(CCCC1)CCC(=O)N2.C(=O)(CCN(C(C)(C)C)C(=O)C=CCO)OC C(=O)(CCCN=[N+]=[N-])NC1(C)CCN(C(c2c(OCC)ccnc2)=O)C1 c1(OC)ccc2c(c1)C(C(=O)NC(C)CCNC(C1(C(=O)OC)COC1)=O)CC2 N1(C(CC(C)(C)OC)=O)CCCC(C)(CNC(=O)Cc2csc(Cl)c2)C1 N1(C(c2n(CC(C)C)ncc2)=O)C2CCC1C(C)C(NC(=O)CN(C)CCO)C2 c1(CNC(c2ccc(C)cn2)=O)nc2c(s1)CCN(C(=O)C(C)OCC1CC1)C2 C1(N(C(c2cc(C(C)(C)C)on2)C(=O)NC2CCC2)C)(CCO)CCCCC1 C1(CC)C(C(=O)NCC(F)(F)C(N)=O)CCCN1C(c1cnc[nH]c1=N)=O N1(C(C(C)=CC2CC2)=O)CCN(C(C2(F)C3CCCCC23)=O)C2(CCC2)C1 CC12CC(C(=O)NC3CCN(C(=O)CC4CC5CC4C5)C3)(C1)C(C)(C)O2 N1(C(C(CC)O)=O)CCN(C(c2cc(C)ncc2Br)=O)CC1CCOC CCCC(C)CC(=O)NC(C1CCCN1C(C1CCC(C)(O)CC1)=O)C C1(S(N)(=O)=O)(CC2CN(C(CC(=O)NC)=O)C2)CC1.n12cc(nn1)C2(C)C C#Cc1ccc(C(=O)NC2CN(C(=O)C(C)c3ncco3)C2)cc1Cl C1(C(N(CCCOCC)C)=O)CN(C(c2c(O)cccc2F)=O)CC12CC2 c1(OC(COCC)=O)c(C)c([N+](=O)[O-])n(C)c1C.C12C(OCCOCC)C1CO2 O=C(NOCCCF)C(C1CCCO1)NC(C1CC2CC2C1)=O C1(C(N(C)CC2CCCN2C(c2ccc(F)s2)=O)=O)CCOC(=O)N1 N1(OC(c2cn3cc(Br)ccc3n2)C)CC2CN(C(C3CC(C)C3)=O)CC(C1)O2 C1(NC(C(CC=CC)NC(=O)CC2CCCC3CC23)=O)CC2C(O)C(O)CC12 CCCC(C(=O)OC)C(=O)NC1CC(NC(=O)C(O)Cc2cn(C)cn2)C1 c1(COC)ncsc1C(=O)NCCC(C)N(C)C(C1CCCCO1)=O Cc1cnc2n1CCC(C(=O)NNC(=O)N1CCN(CCCC(=O)O)CC1)C2 N1(c2nc(C(N)=O)nc(N)c2N)CCC2(C1)OCC1CC21 CC1CC(C(=O)N2CC(C)(CO)C2)=NO1 C(C)(C(C(=O)NCCn1cc(CO)cn1)C(C)C)NC(CCCNC(C)=O)=O C(=O)(CC(CC#N)c1ccccc1)N1C(C)CC(NC(c2[nH]ccc2C2CC2)=O)C1 C1(O)(CN(C(c2c(C)csc2)=O)C)CCCN(C(C2CCNC(=O)C2)=O)C1 CC12CCOC(C(=O)NCC(F)CNC(c3ccnn3CC(F)(F)F)=O)(C1)C2 c1(CC)cc(F)ccc1C(N1CCC(NC(C2CCCCC2)=O)C(CC)C1)=O Cc1ccc2ncccc2c1C(N1CC(OCCNC(=O)C2=CCCC2)C1)=O C1(O)(C(C)NC(CCC#CC)=O)CCN(C(C2CC2c2ccoc2C)=O)CC1 C1(C(=O)Nc2c(C)n(C3CC3)nc2)CCC2CCC1N2C(c1cnsn1)=O c1(NC(CCSC)C)ncc(S(=O)(=O)NC(c2ccc(F)c(C)c2)CO)cc1Cl CCCCC(O)C(C)C(=O)N1CCC(F)(C(=O)NC2CC23CCCC3)C1 c1(C(N(CCCC)CC(N)=O)=O)cc(OC)cc(C(F)(F)F)c1 N1(C(C=CC=CC)=O)CC2CCN(C(c3cccc(F)c3O)=O)CC12 Cn1cc(C(=O)NCC(F)CNC(C2SCCCS2)=O)cn1 N1(C(Cc2c(C)nc(C)s2)=O)CC2(CCN(C(=O)C=Cc3cccc(O)c3)C2)C1 c1(C(N2CC(c3cn(C(C(=O)OCC)C)nn3)C(O)C2)=O)ccc(F)cc1SC c1(-n2c(C3C=CCCC3)nc(CC(C)OC)n2)ccc(Br)cc1C C(C)(CO)(CC(F)F)N(C(c1cc(OC)ns1)C(=O)NCCOC)C Cc1cnn(CC(C)NC(C2CCC(NC(C3CCN3C)=O)C2)=O)c1 CCC(CN(C)C)CC(=O)N1CCC(N2CCC(NC(=O)C(C)(C)C)CC2)C1 CC(C(=O)OC(C)(C)C)C(=O)NCC1CCC1NC(=O)Cc1sccc1Cl C(=O)(CCCCC(=O)N1CCCC(CNC(=O)Cc2ccn(C)n2)C1)NC Cc1cc(N2CCN(C(C3C(C)OC(C)C3C)=O)CC2)n2nncc2n1 N(C(=NCCNC(=O)C(F)(F)F)NCC1=CCOCC1)CC1C(C)(C)CCO1 Cc1cc(CC(N2CCC(NC(=O)Cc3ccc(F)cc3)CC2)=O)n(C)n1 C(=O)(CCCCNCCN(C)OC)NC(CSCCCC)C(=O)NC C1(NC(C(CC)CC)=O)CCC2(CCCN(C(=O)Cc3cncnc3)C2)C1 Cc1ncc([N+](=O)[O-])cc1NC1CCCC1CCCF CC1CN(C(C2CC3C=CC2C3)=O)CC1NC(c1ccccc1C1(C)CC1)=O C(N=c1nc(-c2ccsc2)c(F)c[nH]1)C1CC(NC(=O)Cn2cc(CO)nn2)C1 c1(C(N2CC(O)(C(C)NC(CC=C=C)=O)C2)=O)cn(C)nc1C1CCCCC1 CCC(CC(F)(F)F)C(=O)N(C)CCOCCN(C(=O)CCC1=CCCCC1)C c1(C(=O)OC)cnc(C)nc1SC(C)(C)C.C123CCN(CC1C2)C(=O)N3 C1(CC(=O)NCCC2CCN(C(c3cc(OCC)cs3)=O)C2)(CC=C)CCCC1 C1(C(=O)NCC2N(C)CCN(C(C(C=C)(C)C)=O)C2)CNC(=O)C(C)(C)C1 N=c1[nH]c2c(s1)CCCC2C(=O)NCC(F)CNC(c1ccn2c1CCCC2)=O Cc1cccc(F)c1C(=O)N(C1CCCN(Cc2nnc(C3CC3)o2)CC1)C N1(N(c2cc(C=O)[nH]n2)C)CCC(CCO)(OC)C1.c1(C=O)cocc1C(N)=O C(=O)(CN=c1[nH]c(=NCc2c(F)cc(Cl)cc2F)c2ncccc2[nH]1)NC Cc1cc(=NCc2c(F)cc(F)cc2F)[nH]cc1S(=O)(=O)N1CCN(C)CC1C C(=O)(C1=CCCSC1)NCc1cccc(C(N2C(CC(C)C)CCC2)=O)n1 C1(C(N2CCC(N(C(=O)C=C(C)C3CC3)CC#C)C2)=O)CCn2nnnc2C1 N1(C(CCC(=C)C)=O)CC2(C1)C(NC(C1CCCC3C1C3(F)F)=O)CCS2(=O)=O c1(CNC(CC2(C)CCC2)=O)ocnc1C(N1CC=CCC1)=O N1(C(=O)CC2CCC=CCC2)CC2CC1CN2C(=O)COC1CCC1 CC1CN(C(C2CCCC2)=O)CCC1C(=O)NC(C)CC1CCCCC1 c1(C(=O)NCC=CCNC(C(C)OC)=O)cc2c(nn1)CCCO2 C1(NC(CCC(C)NC(=O)CCn2cnc(=N)[nH]2)=O)(CO)CC2(CCC2)C1 c1(C(N2CC(C)C(NC(=O)C=CC(=O)NC3CC3)C2)=O)cncc2cccnc12 N1(C(c2c[nH]c(=N)s2)=O)CCCC2(CCCN2C(C2CC3CC3C2)=O)C1 N1(C(C2CCN(C(c3[nH]cc(C)c3)=O)C2)=O)CCOC(CN=[N+]=[N-])C1 c1(SCCC(=O)NCCN(C(=O)C(c2ccc(O)cc2)=O)C)ccccc1Cl Cc1cnc(Cl)c(C(=O)N(CCCCN(C(=O)C(C)CC(N)=O)C)C)c1 C=CC(C)(O)CC(=O)NC(C)CC(N1CCC(OC2CC2)CC1)=O C#Cc1ccc(NC(=O)Nc2cc(Cl)c(Cl)c(Cl)c2)nc1F C12(C(=O)NCC3OCCN(C(COCCOC)=O)C3)CCCC(CO1)C2 C(CCN(C(=O)Cc1cc(C)[nH]n1)C)(C(C)(C)C)NC(C1C(OCC)C1C)=O CCC(C(=O)NCC(C1CC1)NC(c1oncc1C)=O)C(C)C C1(NC(C2CC3CCC2O3)=O)CN(C(C2(CCF)CCC2)=O)CCC1C(F)(F)F N1(C(c2cc(SC)oc2)=O)CC2CC2(C(=O)NC2CCN(C)C2=O)C1 c1(C(C(=O)NCC=C)N(C)Cc2cccc(OC)c2F)nc(Br)ccc1OC C1(NC(c2c(C)snc2)=O)CCN(C(=O)CCc2cncnc2)C12CC2 C1(C(N(C(C)(CNC(C2CC(O)CN2C(N)=O)=O)C2CC2)C)=O)CCCN1N=O C=CCCC(C(=O)N(C)CC1CCCN1CC)NC(C1CCCC2(CC2)C1)=O C1(CC)C(NC(=O)Cc2cc(C)[nH]n2)CCN1C(c1cc(C(C)C)n(C)n1)=O Cn1cc(CC(=O)NC2CC(C(C)(C)NC(c3cccs3)=O)C2)cn1 c1(NC(Cn2c(C(C3C(C)(C)C3)N3CCCC3)nnn2)=O)cncc(F)c1 C1(C(C)NC(c2nc(OC)oc2)=O)CCCCN1C(=O)CCCCN(C)C(C)=O Cc1ccc(CC(C)NCC(=O)NC2(C3CCCCO3)CC2)s1 c1(CNC(C(C)OCC)=O)ncoc1C1CN(C(c2nc[nH]c2C(C)(C)C)=O)C1 C=C(F)C1(CC(=O)N(C(C)CNC(c2cc(C(C)CC)no2)=O)C)CCC1 N1(C(CC=CCC)=O)CCC(CCNC(=O)Cc2cc(C)on2)C(F)(F)C1 c1(CCCC(=O)NC(CC)(C)CNC(=O)C(C)CC2CCC2)ccc(C#N)cc1 c1(C(=O)NC2C(NC(=O)Cc3ccsc3)CCC2)cccn2cncc12 Cc1c(C(N2CC3CC3(NC(=O)COc3cccc(F)c3)C2)=O)ccn1CCO N1(C(c2c(CC)onc2)=O)CC2COCC2(C(=O)N(CCF)CCOC)C1 c1(C(=O)NC(C2CCN(C(COCC)=O)CC2)C)ccc(C#N)c(Cl)c1 Cc1cc(C)c(C(=O)NCC2CC3(CC3)CN2C(=O)Cc2n[nH]c(C)n2)c(O)n1 c1(CNC(CC)=O)nc2c(s1)CN(C(=O)C(c1ccc(F)cc1)=O)CC2 S(=O)(=O)(c1ccc(NCc2nc(C)n3ccccc23)cc1Br)NCC(CCC)C c1(NC(C)=O)ccc(CN2CC(C(=O)O)CC2=O)cc1.c12ccc(cc1)c(=O)[nH]2 Cc1c(CNc2cn(C)c(C(=O)Nc3ccc(Br)cc3F)n2)ccnc1Cl N1(C(c2onc(C)c2C)=O)CCCN(C(c2ccco2)=O)C(C(C)C)C1 C(=O)(C1Cc2cccc(Cl)c21)NCCC1CCN(C(CSCC(C)C)=O)CC1 C1(CNC(COCCCCC)=O)CCCCN(C(=O)Cc2cccc(C)c2)C1 C(=O)(C#CC1CCCCC1)N(C1CCN(C(c2c(COC)cc[nH]2)=O)C1)C C1(C(N2CC3C(NC(CC=C=C)=O)(C3)C2)=O)CCCCC(F)(F)C1 c1(NC(CSc2ncc(C(=O)NCC(C)OC(F)F)s2)=O)ccc(F)cc1 C1(C(=O)NCC(C2CC2)OC)CCC(C)(C)N(C(=O)C=C2CCC2)C1 C1(C(N2CCCCC2CCc2cn(CCOCCO)nn2)=O)(CC)CCC(O)CC1 C1(C(=O)NCC(COC)(C)O)C2CCN(C(C3(OC)CC3)=O)CC12 c1(C(=O)NC2CC(NC(C3C(OC)CCCC3)=O)C2)cccc(Cl)c1C(F)(F)F c1(C(=O)NC(CN(C(c2c(Cl)cc(C)c(N)c2)=O)C)C)cccc(Cl)c1[N+](=O)[O-] Cc1cc(=NCC2CN(C)C2)[nH]cc1S(=O)(=O)NCc1ccc(Cl)c(Cl)c1 N1(C(c2c(C)oc([N+](=O)[O-])c2)=O)CCC2(CCCC(C(=O)O)O2)C1 c1(CC(N2CC(NC(CCNC(C3C(C)C3)=O)=O)(CO)C2)=O)ccc(CO)cc1 C1(C)(CNC(c2n(CC)cnn2)=O)CCN(C(c2cnc(C(N)=O)cn2)=O)C1 C(=O)(C1=CCc2ccccc21)N(C)CC1N(C(C(C(C)C)SCC)=O)CCC1 c1(CC(N2CCC(NC(C3CC(OC)C(OC)C3)=O)C2)=O)nsc2ccccc12 CC1CC(CC(=O)N(C2CC3(CC3)C2)C)CN1C(=O)CCCCN(C)C c1(CC)ccc(C(N2CCC2CNC(C2(C(N)=O)CCC2)=O)=O)cc1CC CCCCCC(O)CC(=O)N(C(C)CNC(c1cccn(O)c1=O)=O)C Cn1ncc2cc(CN3CCC(C(=O)Nc4ccc(Br)cc4C(=O)O)C3)ccc12 CC1(C)C(NC(=O)C2=CCCS2)CC1CNC(=O)CCC1OCCO1 c1(CC(=O)NCCCC(C)NC(Cc2c(C)noc2)=O)cn2c(n1)CCCC2 C1(CNC(c2nc(C)sc2)=O)COCCN1C(c1cncs1)=O C1(C(N2CCC(CCC(=O)NC(CC(=O)OC)C)CC2)=O)CC(C)CC(C)C1 N1(C(c2c(C)nsc2C)=O)CCC2(CC1)CC2C(N1CC2(CNC(=O)N2)C1)=O C(=O)(C(C)S(=O)(=O)C(C)C)NCC(CC)NC(=O)C=Cc1ccc(SC)cc1 C1(NC(c2c(C)nc(C)o2)=O)CC2CC1N(C(=O)C=Cc1nc(C)cs1)C2 C1(C(=O)NCCN(C(=O)CCN2CCC(F)C2)C(C)C)(CO)CCOC1 c1(CN2CCCC(C(C)NS(CC)(=O)=O)C2)c(F)cc([N+](=O)[O-])cc1F c1(CC)c(C(=O)N(CCCn2cc(C3(NC=O)CC3)nn2)C2CC2)nnn1C C12(NC(=O)COc3ccccc3)CC1CN(C(=O)CSc1n[nH]c(O)n1)C2 C1(C(C)NC(=O)C(=O)NC(c2ccoc2)C)CCC(C(F)F)CC1 c1(C(N2CC3CC3(C(=O)NCCc3ccc(O)cc3)C2)=O)cccc(Br)c1Cl N1(CCC(C)NC(=O)Nc2nc(C3CC3)nn2C)CCN(C)CC1 C(C(C)(C)CC1CNC1)NC(=O)NC(C)(C)C.C1(C)(N(C)C(=O)OCC)CC1 C1(C(=O)NCCOCCN(C)C(c2ccoc2Cl)=O)C(F)(F)C12CCC2 n1(CC)cc(CN(C(=O)CC2CCCN2C(c2cnsc2C)=O)C)cn1 CCC(C)CCCCC(=O)NCCC(O)CNC(=O)C1=CCCS1 c1(C(=O)NCCCC(C)NC(CCC=C(C)C)=O)cccc(C(=O)OC)n1 c1(NCc2nnn(CC)n2)ncc(S(=O)(=O)N(CC(C2CCCC2)O)C)cc1Cl CC1(C)CN(C(c2cccc(Cl)c2)=O)C(CNC(=O)CC2OCCO2)CO1 C1(CCC(N2CC(N(C)CC)C2)=O)CCN(C(C2CCC2C(F)F)=O)CC1 C#Cc1cc(C(=O)NC2CCC(NC(c3c(C)cccc3Cl)=O)C2)cc(N)c1 C(N=c1nc(C)[nH]cc1C#N)C1OCCN(S(c2ccc(NCC)cc2)(=O)=O)C1 C=CCCC(C)(C)C(=O)N(C)CCOCCC(=O)NCCC(C)N(C)C C1(NC(CNC(=O)NCCCC2CN(CC)C2)=O)CC2CCC(C1)N2C(=O)NC C#CCC(C)(C(=O)NOC1CCCC1)NC(C1C2CCCCC12)=O c1(NCC(C(C)C)N2CCCC2)cc(NCCC(C)(C)c2ccccc2)ncn1 c1(OC)ccc(C(N2CCC(C)(CNC(=O)C(C3CC3)OC)C2)=O)cc1C(C)C C1(C(=O)NCC(CNC(c2ccn(CCF)n2)=O)CO)(CC)CC1(F)F c1(C(=O)OC)cccc(C(=O)NCCN(C)C(C2CC(F)(F)C2)=O)c1C N1(C(c2scc(C)c2)=O)CCc2cc(C(N3CCCC(C(N)=O)C3)=O)ccc2C1 C(CCCC(=O)N1CCCC(CCF)C1)NC(c1n[nH]cc1Cl)=O C(C(C)CC(=O)NC1CCCCC1CNC(=O)Cc1csc(S)n1)OC C(=O)(C1=CCC2CCC1N2C(=O)C(C(C)C)SC)NCC=CCCC N1(C(C2(c3cccc(OC)n3)CC2)=O)CC2CC1CN2C(=O)Cc1occc1C CC(O)(C(=O)NCCCC(c1ccccc1)NC(C1CC2(CC2)C1)=O)C1CCC1 N1(C(c2c(C)ocn2)=O)CCC2C(C1)CN2C(=O)C(C)CSCc1ccccc1 C(=O)(C(CCCC)NC(c1ccc(C(F)F)o1)=O)NCC(CCC=C)O c1(N2CCCC(c3ccc(CC)cc3)C2)nc(NCCC(N)=O)c2ncsc2n1 CC1(C)CCC2(CC1)CC2C(=O)NCC(F)(F)C1CC1 C1(F)(NC(c2cc(CNC(=O)Cc3ccco3)ncc2)=O)CC12CCCCC2 C1(C(=O)NCC(C)(C)NC(C(N2C(=O)CCC2=O)C)=O)Cc2nnsc2S1 c1(C(C)NC2CCCN(c3c(OC)cccc3)C2)cc([N+](=O)[O-])ccc1Cl N1(C(CCC2N(C(c3ncn(C)c3)=O)CCC2)=O)CC(O)C(O)C1 Cn1c(Br)cnc1C(F)(F)C(=O)NC1CCCC1c1ccc(Cl)cc1 N1(C(c2c(OC)csc2)=O)CCC(C)C(NC(=O)C(F)(F)Sc2cnn(C)c2)C1 c1(C(N2CC(NC(c3ccc(CC)cc3)=O)C3C2C3)=O)cc2c(=O)[nH]ccn2n1 C1(NC(C2C(CC)C2)=O)CCCC(NC(c2ccn(-c3ccc(F)cc3)n2)=O)C1 c1(CCNC(CN(C(C=CC(CC)C)=O)C2CC2)=O)ccnc(C)c1 CCCCC(C)(F)C(=O)NC(CC(=O)N1CC2CC2C2CC12)C(F)F Cc1nocc1CC(=O)NC(C1CCN(C(c2ncsc2C(C)C)=O)C1)C C1(NC(C2(C)C(C)(C)C2)=O)C=CCC(C(=O)NCCc2cocn2)C1 CCC(CC(=O)NC(Cc1cn[nH]c1)C(=O)NC(C)C(C)SC)SC CCC(C)(COC)C(=O)NC1CCN(C(C2COCCN2CC(F)F)=O)CC1 c1(C(=O)NC(C)CC2CN(C(C3CCOC3)=O)C2)csc(C(C)(F)F)n1 C1(CCNC(COC(CC)(C)C)=O)CCCN(C(c2cnc(O)nc2O)=O)CC1 N1(C(C(CC#C)C)=O)CC(NC(=O)C#CC(C)(C)C)C(S(C)(=O)=O)C1 C1(CC(=O)NCC(C)(C)OCC(=O)NCC2(N(C)C)CC2)CCC2CC12 c1(C(=O)NCCNC(C2CN(C(=O)C3=CCCS3)CCO2)=O)ccc(O)c(O)c1 c1(C(=O)NC2(CNC(C(C(CC)C)O)=O)CCCCC2)cccc2sccc12 N1(C(c2c(CC)nn(C)c2)=O)CCCCCC1C(=O)NC1CC(C(N)=O)C1 C1(CC(N2CC(O)(CNC(C(C)CC3CCCC3)=O)C2)=O)CCCC2(CCC2)O1 N1(C(CSCCOC)=O)CC(C)N(C(=O)C=CCC2CCOCC2)CC1C c1(C(N2CCN(C(C3C(=C)C3)=O)CC23CCC3)=O)cnc2ccccn2c1=O CC1CN(C(c2ccccc2)CN2CCOCC2)c2ccccc2N(C)C1 c1(C(CNC(c2csc(C(C)(C)C)n2)C)O)ccc2ccccc2c1 C=C(C)CC(C(=O)N1CCN(C(c2cncc(F)c2)=O)C(CF)C1)NC(C)=O Cc1ccc(OCCCC(=O)Nc2ccc(C)c(I)c2)c(O)c1 Cn1ncc2c(O)cc(C(=O)NC3COCC3n3cccn3)cc12 CC(F)(F)C(F)(F)CC(=O)NC(C1CCCC1)CNC(=O)C1=CC2C=CC(C1)C2 CC(CNC(c1ncccn1)=O)CC(=O)NC1CCCN(C)C1 CCCCCCC(CC)C(=O)NC1CC(NC(=O)C=Cc2ccc(Cl)cc2F)C1 S(=O)(=O)(c1cccc(S(=O)(=O)N2CCCC2)c1)N1CC(C)C(C(N)=O)C1 CCCC(CC(C)C)C(=O)NC1CCN(c2nc3cccc(C)c3s2)CC1(C)C Cc1cc(C(=O)NC2CCC(CCC(=O)NCC(O)CC3CCCC3)C2)[nH]c1C c1(SC)cc(C)ccc1C(N1CCC(CNC(=O)C(C)OC2CCCCC2)C1)=O c1(C(=O)NC2CN(C(CCSC)=O)CC(O)C2)c(Br)nc2n1CCC2 N1(C(CC(Cc2c(OC)cccc2)C)=O)CCC2CCN(C(=O)C=C3CC3)C2C1 c1(C(=O)OC)nsc(=NCC2CCCN2C(=O)C(O)C(C)C)[nH]1 C1(C(=O)NC)CN(C(=O)CC2(C)CCN2C(c2ccc(O)nc2)=O)CC12CC2 Cc1cc(=NC2CN(C(c3ccc4nsnc4c3)=O)CC2C)c([N+](=O)[O-])c(C)[nH]1 C(=O)(C1=CC2CC=CCC12)NCc1ccc(CCNC(c2c[nH]c(=N)o2)=O)cc1 c1(OC)ccc(Br)c2[nH]c(=NC3CN(C(C)=O)C3)sc12 c1(OC)ccc(CCO)cc1C(=O)OCCC(F)(F)Cn1cc(-c2csnn2)nn1 c1(OC)cccc(Cl)c1C(=O)NCC1CN(C(C2CC2Cl)=O)C1 C1(C(=O)OCC)CN(C(=O)NC2CC3CC2CO3)CC12COC2 CC1CNCC(C(=O)NC2CCCC2NCCCN2CCCCC2)C1 c1(C(N2CCN(C(c3csc(Br)c3)=O)CC2)=O)cccn(C2CCC2)c1=O C1(NC(=O)NCC(c2ccccc2)CC)CCN(C)CC1 C1(CC(N2CC(CC(C)NC(=O)CCNC(c3ccoc3)=O)C2)=O)CC1C1CC1 N1(C(C(C(=O)OCC)F)=O)CC2CC1CN(C(C13CC(C1)C3)=O)C2 N1(C(c2csnn2)=O)CCC2CN(C(c3cccc4c3CCC4)=O)C2C1 CCCC(C(=O)N1CC2CCC(CNC(=O)C(CCC)NC(N)=O)C2C1)C(C)C C(C(C)(O)CC(=O)N1CCN(C(=O)COc2ccc(CO)cc2)C(CF)C1)OC C1(N(C(C(N)=O)=O)CCO)CCN(C(=O)Cn2ncnn2)C1 c1(C(=O)NCCCN(C2CCCC2)C(COCC(=C)C)=O)nccnc1N N1(C(CCc2c(OC)cccc2)=O)CCC(NC(=O)CC(C)(C)C#N)CC1C c1(CCC(=O)NCC2CC2CNC(=O)CC2CCCCC2)cccc2c1OCO2 Cc1cc(C(=O)NC(C2CCN(C(c3ccns3)=O)C2)(C)C)cc2c1CCC2 C1(C(=O)Nc2ccnn2CCCO)CCN(C(c2cccc(Br)n2)=O)CC1O c1(C(=O)NCCCN2CCC2)cn2cc(Br)sc2n1.C(C)(=O)N.CO c1(C(=O)NCCCCCNC(C(C)SC)=O)cc2c(Cl)cccc2s1 C(=O)(CCCCCC#N)NC(CCCNC(c1c(O)ccc(SC)c1)=O)C C=C(Cl)CC(C(=O)NC(C)CCCNC(C1(C)CC1)=O)NC(=O)OC(C)(C)C CN1CCN(C(C)(C)C(=O)N2CC(CCNC(C3(C)CC=CCO3)=O)C2)CC1 N1(C(c2ccc(CSC)cc2)=O)CCN(C(=O)C=C(C)C(C)C)C(C)C1C C(=O)(C1=C(C#N)CCC1)N1CC(O)CC(NC(c2cccc(SC)c2)=O)C1 N1(C(c2n(CCC)nc(C)c2)=O)CCCCC(N(C)C(c2cscc2Cl)=O)C1 c1(C(N2CCCC(C(C(=O)NCc3c(C)scc3)C)C2)=O)cnc2n1CCC2 c1(NCc2cc(C)cc(Cl)c2)cc(S(=O)(=O)NC2CCCC2C#N)ccc1C#N N1(C(C2C(OC)CCC2)=O)CCC2(CC1)CCN(C(=O)Cc1cc(C)n(C)n1)C2 C1(NC(=O)C=CCN2CCCC2)CN(C(C2CC2F)=O)C2(CCCC2)C1 N1(C(C(C=C)(C)C)=O)CCC2(CCN(C(=O)Cc3cc(F)ccc3Br)C2)C1 C1(NC(C2C(C)CC2)=O)(CO)CCN(C(c2cocn2)=O)CC1 c1(C(C)=O)c(NC(C2(C)CCN(C(c3cnc(O)cc3O)=O)C2)=O)cccc1F C1(C(N2CC3CCCC2C3CNC(C2(CF)CCC2)=O)=O)COCC2(CCC2)O1 CCC(O)CC(=O)N1C(C(N2CCOC(C(N)=O)C2)=O)CC2CC12 C1(S(N)(=O)=O)(C(N(CCCn2cc(C3(C(=O)OC)CC3)nn2)C2CC2)=O)CC1 CC(CC=Cc1ccccc1)C(=O)N(C=O)CC.N1(CC)CC(OC)CC1=O c1(NCC(C)Cn2cccn2)ccc(S(=O)(=O)NCC(CO)C2CC2)cc1Cl N1(Cc2cc(C)c(Br)cc2)CC2CC(CN(C(=O)C(C)(C)CCl)C2)C1 c1(C(=O)NCCN(C(C)C)C(c2ccoc2Cl)=O)noc2c1CCCC2 C(N=c1nc(NCCCCS(N)(=O)=O)c2c([nH]1)c(C)nn2C)c1nc(C)c(C)o1 c1(OCCC(=O)NC(CNC(C(C)OCC)=O)CC(C)C)ccccc1[N+](=O)[O-] Cn1c(O)nc(NC2CN(C(C3Cc4ccncc4C3)=O)CC2(C)C)cc1=O c1(NC(C2CC3(C2)CN(Cc2cocn2)C3)=O)ccc(F)c(Cl)c1F N1(C(C(C(C)O)(C)C)=O)CCC2(CC1)CC(NC(C1(C)CC3CC3C1)=O)C2 C1(C(=O)NC2C(C)COCC2)CC2CCC1N(C(c1cnn(C)c1)=O)C2 c1(N2CC(CC(C)NC(C(CC)(C)OC)=O)C2)ncc2c(n1)CCCCC2 c1(C(N2CC(O)(CNC(=O)CN3CCC(F)(F)C3)C2)=O)cc2ccncc2[nH]1 c1(NC(C2N(C(=O)NCCOC(C(=C)C)=O)CC2)=O)ccc(SC)c(C#N)c1 N1(C(CNC(=O)OCC)=O)CC(O)(CNC(c2cc[nH]c2C)=O)C1 c1(CCCC(=O)NC(C(C)C)C(C)NC(=O)Cn2ncnn2)cc(F)ccc1F C(=O)(CCCC(=O)NCCC1CN(C(C2CC(OC)C2)=O)CC(C)O1)NCCC N1(C(C=CC=CC)=O)CCC2(CCCC2C(N2CCC(F)C(F)(F)CC2)=O)C1 C1(CNC(C(CCC)O)=O)CCN(C(C2CCC(F)C2)=O)CCC1(F)F n1(CCC(=O)NCCCCN(C(c2n(CC)ncn2)=O)C)nc(C)nc1C S(=O)(=O)(c1c(Cl)cccc1Cl)NC(C1CN(Cc2cc(Cl)ncc2C(F)(F)F)C1)=O C1(NC(C(C2CCN(C(C3(COC)CC=CC3)=O)C2)F)=O)CCN2CCC1C2 C(=O)(C(CCC)OC)NCCCC(=O)NC1(C#C)CCC1 Cc1cc(=NC(=O)C(=O)N(CC(F)(F)Cl)C)[nH]n1-c1ccc(F)cc1F N1(CCOC)C(=S)C(c2cccc(C(=O)O)c2OC)NC1C(=O)O c1(OC)nc(Br)cnc1NC(C1CCC(NC(c2cc(C)no2)=O)CO1)=O C1(C(N2CC(NC(CN(C(COC)=O)C)=O)C(C)C2)=O)CCC2CC2CC1 c1(C(=O)NCC2OCCC(NC(=O)Cc3ccon3)C2)ccc(Cl)c2ncccc12 C1(CNC(C2C(NC(C(COC)OC)=O)C2(C)C)=O)COCCOCC1 C1(NC(CCCCC)=O)CCCC12CN(C(C1CCCN(CC(F)F)C1)=O)C2 C1(NC(C(C(C)C)OCC(C)C)=O)CCCCN(C(c2cc(N)cc(F)c2)=O)C1 C(=O)(CCCC(C)(C)NC(=O)Cn1cc(CO)nn1)NC1C(C)COCC1 c1(C(=O)NC2C(NC(=O)Cc3cccnc3)C2)cnn2cccnc12 N1(C(COc2c(C)ccc(C)c2)=O)CCCC2C(CCCN2C(=O)C=CCF)C1 C12(C(N(C3CCC3)C)=O)CCC(NC(c3nnsc3N)=O)(CC1)C2 C(=O)(C1=CC(C)(C)C1)NCC1CC(C)N(C(c2n[nH]c(C3CC3)n2)=O)C1 C1(C(N(CC(C)O)CCNC(C=CCOCCOC)=O)=O)CCOC1(C)C c1(C(=O)NCC(n2cc(CCC3CCCCO3)nn2)C)cc(F)cc2[nH]ncc12 Cc1cc(N)cnc1C(N1CCC(OCC(=O)N(CC(O)C2CC2)C)C1)=O C1(NC(C(CC(C)C)OC)=O)CCC2(CC1)CN(C(=O)CCC(C)SC)CCO2 C(=O)(CS(=O)(=O)C(C)C)NCC1N(C(c2c(F)ccc(CC)c2)=O)CC2(CC2)C1 Cc1c(C(=O)NC(C)CNC(=O)C(F)=C2CCC2)ccc2ccccc12 CCCCCC(O)CC(=O)N1CCC2(CC2NC(=O)Cc2nc(C)c(C)[nH]2)C1 N1(C(C(CC)N(CC)CC)=O)CCC(C2CC2)(CNC(=O)C(C)(C)C(F)(F)F)C1 C(=O)(C1=CC2CCCC12)NC1(C2CN(C(c3c(N)cc(F)cc3)=O)C2)CC1 N1(C(C(C2(O)CCC2)NC(C(C)NC=O)=O)=O)CC2(CCC(C)OC2)C1 n1(C(C)C)cnc(C(=O)NCC=CCC(=O)NCC2CCCCO2)c1 CC1(C)CC(C(=O)NC2COC3(C2)CN(C(=O)CC2=CCCC2)C3)CC(C)(C)O1 C(=O)(C(O)C(F)(F)F)NCC(CNC(C1(CF)CCC1)=O)OC c1(C(=O)NCCC(C)N(C(c2cc(C)c(O)nn2)=O)C)ccc(F)c(C)c1Cl c1(CC)nocc1C(=O)NC1(C)CN(C(c2ncsc2Br)=O)C1 S(=O)(=O)(c1ccc(NCC(C)CCCO)nc1)NC(CCOC)C Cc1noc2cc(NC(C3CCCC3NC(=O)C(C)S)=O)ccc12 c1(NC)cc(C(=O)NCC2(C)CCN(C(c3ccnn3C(F)F)=O)C2)ccc1F c1(CC)ccc(O)c(C(N2CCC(NC(c3csc4cncn34)=O)C2)=O)c1 c1(C(=O)NCC(C)N(C(=O)CC2CCC(C)C(C)C2)C)cccn2nnnc12 C(=O)(C(O)CC(F)(F)F)NC1C(C)CN(C(=O)C(C)(C)C#N)C1 C1(CC)CCN(C(c2cnn(CCNC(C3(C)CCCCC3)=O)c2)=O)CCO1 Cc1c(C(N2CCC(CNC(=O)CSCCC(C)C)C2)=O)cccc1CO Cc1nc(CO)oc1C(=O)N(CCCNC(=O)C(C)NC(C)(C)C)C N1(C(Cn2c(C)ccn2)=O)CCN(C(C2CCC(C)CC2)=O)C(C)CC1C C1(C(N)=O)CN(C(C2(F)CCC2)=O)CCC1NC(c1sccc1CC#N)=O C1(C)(NC(C2CC(SC)C2)=O)CCN(C(=O)C=CCn2cncn2)C1 n1(C(CC)C)ccc(=NC(=O)C2=CCN(C(C3CC4(CSC4)C3)=O)C2)[nH]1 Cc1ccc(C)c(OCC(=O)N(C)CC2(C)CCCC2NC(c2csnn2)=O)c1 C1(CNC(c2cnc(OCC)nc2)=O)CCN(C(=O)CCc2ccco2)CC1C Cc1cccc2[nH]cc(C(=O)NC3CC4CC(NC(=O)CC(=O)N(C)C)CC4C3)c12 N(C1CN(C(=O)Cn2cc(C(C)=O)nn2)CCc2ccccc21)C(C=C)=O CN1CC(N(C(=O)C(C2(C)CC2)NC(c2occc2C2CC2)=O)C)CCC1=O C(=O)(C(C)(CC)C(N)=O)NCC1N(C(c2ccc(CCC)c(N)c2)=O)CCCC1 c1(C(=O)OC)c[nH]nc1C(=O)NOCC(=O)NCCc1ccn(C)n1 CCC(C)C(O)CC(=O)N1CC2C(C(N3CC(C#N)C4(CCC4)C3)=O)C2C1 C1(CNC(C2(CC)CCC2)=O)CC(C)(C)CCC1NC(c1cnc(O)cc1C)=O C1(CC(=O)NCCCCCNC(=O)CSc2nncn2C2CC2)CCCCC1O C1(F)(CNC(C2C(C)(C(=O)OC)C2)=O)CC(NC(C2(N3CCCC3)CCC2)=O)C1 Cn1c(CCNC(C2CCCN(C(=O)C3CC3)CC2)=O)nc2ccccc12 c1(CNC(N(C)Cc2nc(C)on2)=O)ccc2c(c1)C(C)(C)CCC2(C)C Cc1nc(-c2ccccc2)oc1C(=O)NC1CN(C(C2(CF)CNC(=O)C2)=O)C1 C(=O)(CCCN=[N+]=[N-])NC1C(NC(C(=Cc2ccncc2)C)=O)CCC1 CC1(NC(C2CCCCCC2)=O)CCN(C(c2cccc[n+]2[O-])=O)C1 N=c1ccc(C(N2CCCC(CCC(=O)NCC3CC3CO)C2)=O)c[nH]1 c1(C(N2CC3C(CNC(=O)C(c4ccccc4)F)C3C2)=O)cncc2nc[nH]c12 C(N=c1ccnc[nH]1)C1N(C(c2ccnc(Cl)c2)=O)CCOC1 C1(C(=O)NC(C)CCNC(C2CC2F)=O)(C(=O)OC(C)(C)C)CCCCO1 c1(CC)cc(C(=O)NC(Cc2cnc[nH]2)C(=O)NCC2CC(CF)C2)ns1 c1(NC)cncc(C(=O)NCCN(C(=O)C(F)OC(C)=O)C)c1 C1(C(N2CCCCC(CNC(=O)C=CBr)CC2)=O)CCc2nc(O)[nH]c2C1 S1(=O)(=O)C2=CC=CC(=NCCN1)N2.C(C)(C)(CC)CC(=C)Br.C(C)(C)O CC(O)CCC(=O)N1CC2C(CNC(c3cccc(Cl)c3)=O)C2C1 C1(C(=O)NCC2CCC3CC23)(CNC(CCc2cnc(C)o2)=O)CC(C)(C)C1 c1(C(=O)NCCC(CNC(c2c(C)nncc2)=O)O)cnc2c(C#N)cnn2c1 c1(C(N2CCC(C(C)NC(C(CC=C)(F)F)=O)C2)=O)cccc2cccnc12 CC(CCSC1CCN(c2ccc(C(=O)O)nn2)CC1)CC(C)(C)C CC1(C)CC(NC(=O)C=CC2CCCO2)CN(C(=O)CC2CC(F)C2)C1 c1(CN(C)CCOC(C)(C)C)cn(C2C=CCCC2NC(=O)C(F)F)nn1 C1(CCCCNC(C2CCCN2C2CC2)=O)CCN(C(=O)C(F)(F)C2CC2)C1 C=C(C)CCCC(=O)N1CCCCCC1.C1(C)C(=O)N1Cc1nccs1 N1(C(c2ccc(C(=O)OC)nc2)=O)CCCCC(NC(=O)CSC(=N)N)C1 C1(C(=O)NC2C(C)N(C(C3COCCO3)=O)CC2)CCc2n[nH]cc2C1 N1(C(C(F)=CCC)=O)CCC2CCN(C(c3cc(F)c(F)cc3OC)=O)CC12 C(c1cncnc1O)=CC(=O)NCC1C(NC(c2c(OC)nn(C)c2)=O)CCC1 N1(C(C(C)=C2CC2)=O)CCCOC(CCNC(C2CCCCS2)=O)C1 c1(OC)cc(C(=O)NCCN(C(c2ccc(O)cn2)=O)C2CC2)nnc1C1CC1 C1(CNC(CNC(N)=O)=O)CC12CCN(C(c1ccc(Cl)cc1O)=O)CC2 C1(C(=O)Nc2ccc(C(C)(C)C)cc2)CN(S(=O)(=O)C2CC2)CC1(F)F N1(C(C2N(C(C(CC)=O)=O)CCC2)=O)CCC(Oc2ccccc2Cl)CC1 C1(N(C(C2CC(C)C2)=O)C)CCN(C(=O)CC(C)C2CC2)C1 CC1(C)CCC(C)(C(=O)NCC2CCC3(CN(C(=O)C(O)P(C)(C)=O)C3)O2)CC1 c1(C(N2C(CNC(=O)CCSCC(N)=O)CC(OC)C2)=O)ccc(F)c(Cl)c1N CC1C=C(C(=O)NC2CCCCN(C(c3ccc([N+](=O)[O-])o3)=O)C2)CC1 Cc1c(C(=O)NC(CCC#C)C(N2CCC3(CCCC3)C2)=O)cccc1C#N C(=O)(C1=CC(C)(C)C1)N1CCC(CC=C)(NC(=O)CCSCC(N)=O)C1 C#CCCC(O)C(=O)NCC(C)(O)CNC(=O)C=CCN1CCC1 C12(NC(c3c(C)n(CC4CC4)cc3)=O)CCN(C(C3(Br)CC3)=O)CC1C2 N1(C(C(C(C)(C)C)OC)=O)CC2(C1)C(NC(=O)CC1(OC)CCC1)CCS2(=O)=O c1(CC)ccccc1C(CNC(C1C=CCCC1)=O)NC(=O)CN(C)CCOC Cc1nc(C(=O)NCC2CC2NC(=O)Cn2ccnc2C(C)C)ccc1[N+](=O)[O-] C(=O)(C(O)CC(C)(C)C)NCC1(O)CC(C(=O)NCc2c(C)cccn2)C1 c1(CN(C(=O)CN2CCCC2C(C)(C)C)C(N(C(C)C)C)=O)c[nH]nc1[N+](=O)[O-] C1(CCOC)(C(N2CCC(N(CCO)C(C3CCS3(=O)=O)=O)C2)=O)CCCC1 C1(C(=O)NCCc2c(C)nc[nH]2)CCN(C(=O)C=CC2CCCC2)C1C c1(COC)cc(NC(=O)CC2CCCC2C)cc2c1OCOC2 C(=O)(C1c2ccccc2OCC1(C)C)NC1CC(NC(CCOCC)=O)C(O)C1 C(=O)(C(F)(F)CCn1cccn1)N1CCC(C)(CNC(=O)Cc2nnc(O)s2)C1 C1(C(N(CCCNC(C2CCCCO2)=O)CC)=O)COc2c(F)cc(F)cc2C1 C1(CN(C(C2CC(=O)N(O)C2)=O)CC)CCCN(C(c2cc[n+]([O-])cc2)=O)C1 c1(C(N(C2CCCN(C(CNC(CC)=O)=O)C2)CC)=O)ccc(OC)nc1C C(=O)(C1=C(C)S(=O)(=O)CC1)NCC1CN(C(CC(=O)NCC#C)=O)CC12CCC2 C12(C(N(C(C)C(=O)NCCCn3nccn3)CCC)=O)CCCN(CC1)C2 CC1C(C(=O)NC2(C)CCCCC2C(=O)NCc2cncc(Cl)c2)=NOC1C Cc1nc(SCC(=O)OCC2CCC3(CCC3)CO2)c(C(N)=O)c(C)c1C CC1CN(C(C23CCC(CC2)C(C)(C)O3)=O)CC2(CCN(C(=O)C(C)C#N)C2)O1 c1(OC)ccncc1C(=O)NC1(C2CCCN2C(=O)C=Cc2ncc(C)[nH]2)CC1 c1(C(=O)NCC2CN(C(Cc3cc(C)[nH]n3)=O)C(C)(C)C2)nc[nH]c2nccc1-2 C(=O)(C(C)CCC(C)(C)C)N1C(CO)CC(NC(C(C=CC)O)=O)C1 c1(NCCSN(c2nccs2)C(=O)COCCCn2cncn2)cccc(F)c1 C(C(C(=O)NCC(n1cc(-c2ncoc2C)nn1)C)OC)OCC N1(CCC)CC(C(=O)NCCC2CCN(C(C34CC(C)(C3)C4)=O)CC2)CC1=O c1(C(=O)NC2C3(CC(NC(c4cnns4)=O)C3)C2)c(F)ccc2ccoc12 CC1(CN2CCC(F)(Cn3cc(CS(C)(=O)=O)nn3)C2)CCCC1(F)F C1(NC(c2nc(C)oc2)=O)CN(C(C2CC(O)CN2C(N)=O)=O)CCC1C C(N=c1nc(C2CCCC2)[nH]s1)C1CN(C(COCc2c(C)ncs2)=O)C1 N1(C(C=NOC)=O)CC(NC(=O)Cc2ccnc(O)c2)C(C(F)F)C1 N1(C(CCC(=O)OC)=O)CCOCC(F)(CNC(=O)Cc2cccs2)C1 Cc1cccc2c1CN(C(=O)C(CNC(c1cc3cc[nH]c3cn1)=O)N(C)C)C2 c1(C(N2CC(C)C(C(=O)NCC(F)Cl)C2)=O)ccc(N)c(F)n1 c1(C(N(CC(C)N(C(COC)=O)C)C)=O)csc2cc(Cl)cnc12 c1(C(C)C(=O)NC(C)(CNC(C2(c3cc[nH]n3)CC2)=O)CO)ccc(Cl)cc1 N1(C(C(CC=C)CNC(=O)C(CCC)NC(C)=O)=O)CCC2(CCC(OC)C2)C1 Cn1cc(S(N)(=O)=O)cc1CC(=O)NCC1=CCSC1 C(=O)(C1=CC2CCCC12)N(CC(CNC(Cc1ccc(OC)c(O)c1)=O)(C)C)C C(=O)(CCCCCN(C)C(C1CC2C=CC1C2)=O)N(C)CCOCC1CC1 N1(C(c2cccc(CC)n2)=O)CCC(C2CC2)C1C(N1CC(C)(C2CCC2)C1)=O c1(CNC(C2N(C(CC3C(=O)NC(=N)S3)=O)CCCC2)=O)ccc(F)nc1F C=CCC(CC=C)C(=O)NC(CCSC)C(=O)NCC1(C2CC2)CC1 c1(N2CC(=C(CNC(CCCC(C)C)=O)F)C2)ccc([N+](=O)[O-])cc1Cl C1(C(=O)NCC(n2cccn2)C)CC(F)CN1C(=O)CCC(C)N(C)C1CC1 c1(CC(=O)NC(C)CCN(C)C(C2C=CCCC2)=O)ccnc(O)c1Br c1(C(=O)NCC2N(C(CNS(C)(=O)=O)=O)CCC2)ccc2nc(Cl)ccc2c1 C12(C(=O)OC)CC1CCCN2C(=O)NCCc1cc(OC)nn1C C(=O)(C1=Cc2ccccc2C1)NCC(CC)NC(c1ccc(Cl)c(OC)c1F)=O c1(CC(N2CCCCC(NC(c3[nH]n(C)c(=O)n3)=O)C2)=O)cnn2ccccc12 c1(CC)nnc2n1CCCC2c1nc(CC)n(-c2cccnc2)n1 C12(CNC(CCC#CC)=O)CC(NC(C3CC4CC3C3CC43)=O)(CCO1)C2 c1(C(=O)NCCCN(C(=O)COC(F)F)C(C)C)cnc2ccc(C#N)cn12 N1(C(CCOc2ccc(C)cc2)=O)CC2(CC(NC(=O)CC3C=CCC3)C2)C1 c1(C(C)C)ncncc1C(=O)NC1CC2(C1)CC2NC(C1CCC(=O)N1)=O C(CNC(=O)Cn1cnc(C#N)n1)(CC(=O)NCC1NC(=O)NC1=O)OC C=CCC(C(=O)NCC(=O)NOCCOC)NC(c1ccccc1)=O Cc1nsc(C(=O)NC2(CO)CCN(C(C3CC(N(C)C)C3)=O)C2)c1N N1(C(C(CCOC)(C)C)=O)CC2(C1)OC1(C)CC2(NC(C2CCCC2(C)C)=O)C1 c1(C(=O)NC2C(NC(C(C(C)C)NC=O)=O)CCC2)cnc2c(c1)N(C)CCO2 c1(C(N(C(C)C)CCNC(=O)C=CS(C)=O)=O)ccc(S(C)(=O)=O)cc1Cl c1(CN(C2CCOCC2)CC)ccc(C(=O)O)cn1.C1C(C)(C)CNC(=O)N1C N1(C(CCc2nc(C)c(C)[nH]2)=O)CCN(C(c2cn(C(C)C)nn2)=O)CC12CC2 N1(C(c2n(CC=C)ccc2)=O)CCN(C(=O)C=COCC)C(C(C)C)C1 C12(C(=O)NC(CNC(c3c(C)snc3)=O)(C)C(C)C)CCCCC(F)(C1)C2 N1(C(=O)NC(C)CC(N)=O)CCCC(C2CCN(C(c3ccccc3)=O)C2)C1 c1(C(=O)NC(CNC(c2cc(COC)cn2C)=O)C(C)C)cnn2ccncc12 Cc1ccc(-n2cc(C3(C(=O)NC(C)(C)CNCCO)CC3)nn2)cc1Cl.NC1CC1 N1(C(c2n(C)ncc2)=O)CC(NC(=O)CCOCC(F)(F)F)C(n2cccn2)C1 c1(C2(C(=O)NCC(CCNC(C3C4CCCOC34)=O)O)CC2)cccc(Cl)c1 N1(C(C(=O)NC(c2ccccc2)C(C)C)=O)CCCC1CCN(C)C C1(CNC(C=CC(=O)OCC)=O)CN(C(=O)CC2C(=O)NN=C2C)CC1OCC CC(C)CC(C)(O)C(=O)N1CCC(CN(C)C(c2cnccc2C(F)F)=O)C1 C1(NC(C(C)OC)=O)CN(C(c2csc(C)c2)=O)CC2(CCC2)C1 Cn1nnc2cc(C(=O)NC3CC(NC(C4CCC(C)(O)CC4)=O)C3)ccc12 c1(SCn2cc(C(C(=O)NC3C(OC)C(O)C3)N(C)C)nn2)ccc(Cl)cc1 c1(C(=O)NCC2CCN(C(CC3CC(=O)NCCC3)=O)C2)[nH]nc([N+](=O)[O-])c1Cl c1(OC)cccc(NC2CN(C(=O)C(C)(C)C3CCCO3)CC2(C)C)c1[N+](=O)[O-] C1(NC(=O)CSc2ccncc2)CCN(C(C2CCCSC2)=O)CC1CO c12ccccc1C(=O)N(C1CCNC1=O)C2.c1(C(C(C)C)O)cn(C(C)C)nn1 C1(CC(=O)NCCC2CN(C(=O)CCn3cncn3)CCO2)CCCNC1=O C1(CNC(C(C)CC2CCCCC2)=O)CN(C(C2(F)CCCC2)=O)CC12CC2 N1(C(c2c(NC)scn2)=O)CC(O)CC1C(N1CCCC(CC2CC2)C1)=O Cc1ccc(F)c(C(N2CC3(CC(CNC(=O)CSC4CC4)C3)C2)=O)n1 CCCCC(CN=c1nc(OC)[nH]c(OC)n1)NC(c1cc(F)c(F)cc1F)=O c1(-n2c(-c3nn(C)cc3C)nc(CC(CC)C)n2)ccc(OC)c(OC)c1 O=C(C1=CC2C=CC1C2)N1CC(C(N2CCCC23CCC3)=O)C2(CC2)C1 C1(CC(=O)N(C2CC(C)(NC(N)=O)C2)C)CN(C(=O)C=C2CCOCC2)CCO1 c1(OC)ccc(NC(=O)C(c2ccc(Sc3ccc(C(N)=O)cc3)cc2)=O)cc1F C1(NC(CC2(COC)CCCC2)=O)CCC2CCN(C(C3CCC=CO3)=O)C1C2 CC1C(O)CCCN1C(c1ccc(NS(=O)(=O)Cc2ccc(Cl)cc2)nc1)=O N1(C(C(C2CC(C)(C)OC(C)(C)C2)F)=O)CCOc2ccc(Br)cc2C1 N1(C(CC(C)N(C)C)=O)CCC2(CC1)COC(CNC(C1C3CC4C(C3)C14)=O)C2 C1(NC(C(C=C)O)=O)CN(C(=O)CCCCc2ccccc2)CC1F CC1(CNC(C2CNC(=O)C2)=O)CCN(C(=O)Cc2csc(-c3ccsc3)n2)C1 C1(CS(=O)(=O)NCC(c2ncccc2Cl)C)CCC(C(F)(F)F)CC1 c1(COCC(=O)NC2CCN(C(=O)C(F)C=CC(N)=O)C2)ccccc1 C(=O)(CCCCCN(C(=O)C=Cc1ccncn1)C)NC(c1cccc(F)c1)C c1(CNC2C(C)CC2)ccc(OCC(F)(F)F)cc1Cl C(CCC(=O)N(C(C)CCNC(=O)COCC1CC1)C)OC(CCC)=O c1(CC(=O)NCC(CNC(C=C(COC)C)=O)C)c[nH]c(=N)nc1O C(C)(CC(C)CC(C)C)(c1n(CC)nnn1)NCCNC(=O)NC(C)C C(=O)(CC1=CCN(C(=O)C#CC(C)(C)C)CC1)NC1C(CC)CCC1 C(CC(=O)N1CCN(CCC(=O)NC(N)=O)CC1C)(C(C)C)CC c1(C(=O)OC)cc(C)nn1C.C1(CNCc2n(CC)nnn2)CCCC1(C)C C(=O)(C(O)CC(C)C)N1CC(C(N2CCC2(C)C(C)C)=O)(SC)C1 CCCC(C(=O)NCC1(NC(=O)CCCn2nc(C)cc2C)CCC1)OC N1(C(C2N(CCC)CCC2)=O)CCC2(CCC2)C(NC(=O)C(=O)N=S(C)(C)=O)C1 Cc1nc(CN(C(=O)CCc2ccccc2)C(C)C)oc1C(=O)O c1(C(=O)NCC23N(C(C4CCN(C)CC4)=O)CC(CC2)C3)onc2ccccc12 c1(C(N2CC(OCC)(CNC(C3(CO)CC(C)(C)C3)=O)C2)=O)nc(C)ccc1C c1(C(N2CC(CNC(=O)CC3C=CCC3)C(O)C2)=O)ccc2ncccc2c1Cl c1(CC)ccc(O)c(C(N2CCC2CNC(=O)CC2(C)CCCO2)=O)c1 c1(NCC2CC3(CC(NC(c4cc(C)no4)=O)C3)C2)cc(=O)n(C)c(O)n1 N1(C(C(c2cnn(C)c2)OC)=O)CC(CO)(NC(C2CCC(CN(C)C)O2)=O)C1 N1(c2cc(NCCn3cnnn3)ncn2)CCC2C(CCCN2C2CC2)C1 C(C)(c1ccco1)=CC(=O)NC(CC=C)CNC(c1cc(OC)cs1)=O c1(C(N2CC(O)(CN(C)C)C2)=O)ccccc1-n1cc(C2(C3CC3)CC2)nn1 CC(C)CC(C(=O)NC(CCC(=O)N1CCC(F)(F)C(O)C1)C(C)C)C(C)C C(=O)(C1=NNC(C(F)(F)F)C1)NCC1N(C(CSCC=C)=O)CC(COC)C1 N1(C(Cc2nc(C)[nH]n2)=O)CCCC(C)(CNC(C2CC3OC2C2CC32)=O)C1 C=CCC(CNC(c1cc(C)sn1)=O)C(=O)NCC(N1CCCCC1)=O c1(C(=O)NCC23N(C(CNC(=O)OC)=O)CCC2CC3)cc2c(s1)CCSC2 c1(C2CNC2)cn(C(C)C=O)nn1.C1(C(C)COC(=N)O)CCCC1 c1(N2CCCC(C=C)C2)nc(=NCc2cc[nH]n2)[nH]c2c(F)cc(F)cc12 C(CC1=CCN(C(c2cc(SCC)cnc2O)=O)CC1)NC(CCOCC)=O N1(C(C2CN(OC)C(=O)C2)=O)C2CC=C(C(=O)NCC3CCC=CO3)C1CC2 N1(C(C=CC2CCN(C(C(CCCC)OC)=O)CC2)=O)C2CCC1CN(C)CC2 C1(NC(C(c2cccnc2)NC(CCCO)=O)=O)CCC(CCO)CC1 c1(C(N(C2CCCC(NC(C3(F)CCOC3)=O)C2)C)=O)nccn2nccc12 CC(C)CC(F)(F)C(=O)N1CCCC(C)C1CNC(C1CCSCC1)=O Fc1c(-c2nc(-c3nc[nH]n3)nn2-c2cn3ccccc3n2)ccc2c1CCC2 N1(C(c2cn(CC)nc2C2CC2)=O)CC2CC(C)N(C(=O)CC3(CO)CC3)C2C1 C1(NC(C2N(C(=O)NC(C)C)CCC2)=O)CN(C(C2C3COCC23)=O)CC1O N1(C(c2ccc(F)cc2Cl)=O)CC2(C1)CN(C(C1CC(O)C1)=O)CCO2 c1(OC)c(Br)ccc(C)c1C(N1CCC2(C1)CN(C(=O)OC(C)(C)C)C2)=O CC1CCN(C(c2ccncc2-c2ccc3c(c2)CCCO3)=O)CCC1(F)F Cc1c(N(C)CC2CCN(C(=O)CN3CCCCC3=O)C2)ncnc1Cl C1(NC(CCC#C)=O)CC=C(C(=O)N2CCC(CC(=O)OCC)C2)C1 c1(C(N2C(C(C)NC(COC(C)=O)=O)CCCC2)=O)cc(C)c(C)nn1 c1(OC)ccc2c(c1)OCC2CC(=O)N(C)C(C)C c1(C(N2CCC(CNC(COCCCCC)=O)C23CC3)=O)cc(N)c(F)cc1C N1(C(=O)NC2CCC=CCC2)CCc2ncsc2C1 N1(C(C2N=C(C)SC2)=O)CCCC(C)(CNC(c2ccc(=O)n(C(C)C)c2)=O)C1 C1(NC(c2cc(OC)n(C)n2)=O)CC12CCN(c1ccnc(C3CC3)n1)CC2 C(=O)(CC(O)CC(C)(C)C)N1C(C(=O)NC(CC)C(C)(C)C)C(O)CC1 c1(OC)ccc(Cl)cc1C=CC(=O)NC(C)CCCNC(=O)C1=NNC(=O)C1 C=C(C(=O)N1CCC(C)(C(=O)NCc2cncnc2)CC1)C(F)(F)F C1(O)(C(N2CCC(C(=O)NCCCN3CCCC3=O)CC2)=O)CC2CCC1C2 CCCC(C)(O)C(=O)N1CCCC(C2CCCCN2C(c2ccoc2Br)=O)C1 CC(c1ccccc1)=CC(N1CCN(C(C2(C(N)=O)CCC2)=O)CC1C(C)C)=O C(N=c1[nH]c(=NCCCC(C)(F)F)c2ccc(C)cc2[nH]1)C1(CC=C)CCCC1 C=CC1CCCN1C(=O)CC1CCN1C(=O)Cn1c(C)ccc1C c1(C(c2n(CCCC)nnn2)NC(C)CCO)n[nH]c(C)c1C C1(C(N(C)CC2CCCN(C(c3cc(Cl)cs3)=O)C2)=O)CCC2(CCC2)CO1 C1(c2cn(CCOC)nc2)(CO)COCCN1C(c1cc(O)cc(F)c1)=O N1(C(CCC=C)=O)CCN(C(c2coc(CO)c2)=O)CC2CCCCC12 CCCCC(CC(=O)N(C)C(c1cnnn1C)C)NC(C1C=C(C)CS1)=O C1(NC(=O)CC2(CO)CCCCC2)CCN(c2ncc(O)cn2)CC1O c1(C(N2CC(OC)C(NC(C3(O)COC3)=O)C2)=O)cc2n(n1)CCO2 C1(C(C)C)CN(C(=O)C(=O)NCC2CC2)CCC1NC(c1cnc(C(N)=O)s1)=O c1(OC)ccccc1C(=O)NC(C)C(CO)NC(C1CC1c1ccncc1C)=O c1(OCC(=O)NCCN(C(=O)Cc2nc(=N)[nH][nH]2)CC)cccc2ccccc12 c1(C(=O)NC23CCN(C(C(=O)N(C)C)=O)CC2C3)ccc2ccnc(O)c2n1 N1(Cc2c(Cl)ccc(OC)c2)CCC2(CCN(C(=O)CNC(=O)C(F)(F)F)C2)C1 N1(C(C2CCN(CC)C2)=O)CC(F)(F)CC1CNC(c1cc(C(C)(C)C)c[nH]1)=O C(C(F)(C(=O)N(C)Cc1occc1C)C(C)C)NC(C1(CC)CCOC1)=O N1(C(C23C(C(=O)OC)(CCC2)C3)=O)C2CCC1CN(C(c1cc(C)c[nH]1)=O)CC2 C1(NCc2cc(C)ccc2C)CCC(NCC(=O)NC(C)=O)CC1C(F)(F)F N1(C(C(C)(C)OCC)=O)CCC2C(CCCN2C(c2cnc(C)c(N)c2)=O)C1 C12(OCC)CCC(C(=O)NCC3CCN(C(c4cc(Cl)ns4)=O)C3)(CC1)C2 C=CC1(C(N2CC(O)(C(F)(F)F)C2)=O)CCN(C(C2CCCCN2CC)=O)C1 N1(C(Cc2c(C)nc[nH]2)=O)CC(O)(C2CCN(C(=O)C=C3CCCCC3)CC2)C1 C#CCC(C(=O)N(CC(=O)Nc1cncc(Cl)c1)C1CCC1)C1CC1 N1(C(C=CC)=O)CCC2(CCN(C(=O)Cn3cc4ncccc4n3)C2)C1 C(c1nc2ccccc2s1)=CC(=O)N(C1CC(NC(c2cc(OC)n[nH]2)=O)C1)C c1(CC)cc(C(=O)NCCC2CC(NC(=O)C(C)CN3CCCC3)C2)ncn1 Cc1cccc(C)c1C(=O)NC1CC2(C1)CC(C(=O)NC(C)C(C)(C)O)C2 C1(C(=O)NCCCc2ccc[nH]2)CC12CCN(CC1CCS(=O)(=O)C1)CC2 N1(c2nc(NCCN(CC)CC)c3c(n2)scc3)CC(C)OC2(CCCCC2)C1 c1(OC)ccnc(C(N2CCC(CN(C)C(C34COCC3C4)=O)CC2)=O)c1OC c1(OC)c(NC(N2CC(n3nc(C)cc3C)(O)C2)=O)cc(C(=O)O)cc1C c1(C(N2CCC(NC)C(C)C2)C(=O)NCc2cccs2)cc2ccccc2cn1 C1(CNC(CCOCCN(C)C)=O)CC2(CCN(C(=O)C(C)C)C2)CO1 c1(C(C)C)nn(C)cc1C(=O)NCC1CCCCN1C(C1(C(C)(F)F)CCC1)=O N1(C(CC2CC(CC)C2)=O)CCCCCC(NC(c2cc(C)c(F)cc2F)=O)C1 Cc1nc2ccc(C(=O)NCC3CC(O)CN3C(=O)Cc3c[nH]nc3O)cc2o1 Cc1nn(CC(=O)NCCCN(C(=O)C(C)C(F)F)CC2CCCC2)c(=O)o1 C1(NC(=O)Cc2cccnc2O)C2CCC(C2)C1C(=O)N(C12CCCC1C2)CCO Cc1nn(C)c2cc(C(=O)Nc3cncc(Br)c3)cnc12.N1CCOCC1 N1(N(c2ccc(NCC)cc2)C(C)=O)CCN(CC)C(=O)C1C c1(C(N(CCNC(=O)C(C)OC2CCCC2)CC)=O)nc2cc(O)ccc2[nH]1 n1(CC)nnc(C(N2CCC(C3CCCCN3C(=O)C3=NOCC3)CC2)=O)c1C c1(OC)ccc(NC(=O)COC(C)(C)CNC(c2occc2Br)=O)c(C)n1 c1(C(=O)NCCC(C)N(C(=O)C(F)CC2CCCCC2)C)cc2[nH]ccc2s1 c1(C(=O)NCC2CN(C(CC(CC)C)=O)CC2C)c(C)nn(CCO)c1C N1(C(C(C)=C2CC2)=O)CC(NC(=O)CCc2ccnc(Cl)c2)C(F)C1 C(=O)(C1=C(F)CN(C(C2(C)CCC3CC3C2)=O)CC1)N(CC)CC1CCC1 c1(C(=O)NCCN(C(=O)CCC(=O)C2CC2)CCOC)ccc2cccnn12 c1(C(=O)NCC2(F)CC(NC(C3(n4cccn4)CCCC3)=O)C2)ccnnc1S C1(NC(C(C)CSC(F)(F)F)=O)(CO)CCCN(C(C2CNC(=O)N2C)=O)C1 CC1CCN(C(c2cccc3cncn23)=O)CCN1C(c1ccc([N+](=O)[O-])s1)=O N1(C(c2nc(C)c(F)cc2)=O)CC2CCC(C1)N2S(=O)(=O)CCc1ccccc1 c1(OC)cccc(-c2nc(C(C)OCC)n(-c3cnn(C)c3)n2)c1.C(C)(C)(C)O c1(NC(C2CC(O)CN2C(c2cc[n+]([O-])cc2)=O)=O)c(Br)cc(F)c(F)c1F Cc1csc2ncc(C(=O)NC(C)(CNC(=O)COC(C)(C)C)C(C)C)n12 NC(=O)CC(O)C(=O)N(C1CCN(C(C2(C(F)(F)F)CC3(CCC3)C2)=O)C1)CCO C(=O)(C(C)(C)CC(F)F)N1CC(C(N2CCC(C=C)CC2)=O)C(C(C)C)C1 c1(CC(=O)NC2CN(C(c3c(Cl)cc(C)s3)=O)CC2C)ccc(F)cc1C C1(NC(=O)C(F)CC2CCC2)CC12CCN(C(=O)CCC1CCCCCC1)CC2 C1(NC(c2cc(C)ncc2)=O)CCCCC12CCN(C(=O)CC1CC1C)CC2 c1(SCC2(C(C)O)CC2)ccc(-c2ccnn2C)cc1OC N1(C(C(CO)N(C)C)=O)CC2CCOC2(CNC(C2(F)CC3(CCC3)C2)=O)C1 Cc1ccc(I)c(NC(C2CC3(CC3)CN2C(=O)CSc2ncccn2)=O)c1 N1(C(C=CC(N)=O)=O)CCC(CCNC(=O)CSc2nnc(S)s2)CC1 C1(C(=O)N(CCC(C)NC(=O)COC2(C)CCC2)C)(OC)CCC(C)(C)C1 N1(C(C23CC(C)C2C3)=O)CC(NC(C2CCCN2S(C)(=O)=O)=O)CC12CCC2 N1(C(C)=O)CCC=C(C(=O)NC2CC2)C1.c12cscc1C(C)(C)N2 N1(C(c2cc(CC)nn2C)=O)CC2CCCC(CNC(=O)C(F)OC)C2C1 c1(CC(=O)NCC(CC)NC(=O)CC2CCC2(C)C)c(F)cc([N+](=O)[O-])cc1F C(=O)(CCS(C)(=O)=O)N(C)CC1CN(C(C2(C(F)F)CCCO2)=O)C1 N1(C(C2OCCC(NC(C3CC4(C3)CC(O)C4)=O)C2)=O)CCC2(CCC2)C1 c1(CC(=O)NC2(C(=O)NCCC(COC)OC)CC2)ccc(C#N)cc1 N1(C(C=CSC)=O)CCC(NC(=O)C=Cc2cc[nH]n2)CC1C CC1(C)CCCc2cc(C(N3CC4CC(NC(=O)Cc5ccon5)C4C3)=O)sc21 C1(C)(C(=O)NCCCOCCNC(C(CCOC)C)=O)CCC12CCC2 C(CN=C(NCc1ccc(C)c(O)c1)N1CCC2(CCOCC2)C1)N(CC)CC N1(C(=O)Cn2ccnc2)CCN(c2ccc(-c3ccc(COC)cn3)cc2)CC1 C1(COC)CN(C(c2cnc(C3CC3)[nH]2)=O)CCN1C(c1ccncc1C)=O c1(NC2(c3nnnn3CCCF)CCCC(C)C2)ccc2cccnc2c1 N1(C(=O)CC2CC(F)(F)C2)CCC(C2CCN(C(C3CN(C(N)=O)C3)=O)C2)CC1 N1(C(C2N(C(C)=O)C(=O)CC2)=O)CC(NC(C2CC2CC(C)C)=O)CC1(C)C c1(C(=O)NCCN(C(=O)Cn2ccc3ccccc23)CC)cnc(Cl)c(F)c1N c1(C(=O)NC(CNC(C(c2nccc(C)c2)(C)C)=O)C)cc(C#N)n(C)n1 C1(C(C)C)CCCN(C(C23CC2CCN3C(c2ncccc2N)=O)=O)C1 CN1C(=O)CSC1=CC(=O)N1CC=CC(NC(C2CCCCC2O)=O)C1 C(C)(C(=O)N=c1cc(C)n(C)[nH]1)N(C(C(C(CC)C)OC)=O)CC N#Cc1ccc(NC(C2CCCCN2C(c2ccccc2C#N)=O)=O)cn1 Cc1cc(NC(c2csc(=N)[nH]2)=O)ccc1NC(C12CCC(CO1)C2)=O c1(C(=O)NCC#CCNC(Cn2ncc(C)c2)=O)cccc2c1CCO2 c1(OC)cc(CN2CC3C(C2)N3C(=O)C(C)(C)F)ccc1C#N N1(C(C#CCNC(c2cnoc2)=O)=O)CC(F)(F)C1C1CC1 Cc1ccc2[nH]c(C(N3CCC4CCN(C(=O)C(F)F)CC34)=O)c(Cl)c2c1 c1(C(=O)NC23C(CN(C(C(C)CN(C)C)=O)C2)C3)ccc2nc(C3CC3)oc2c1 Cc1nc(O)c(C(=O)N(CCNC(c2ncn(C)n2)=O)C2CC2)cc1Br CCC(C)CC(C)C(=O)NCc1cc(C(N2CCC=C(F)C2)=O)no1 C(=O)(C1=C(C2CCCCC2)N(C2CC2)C(=O)NC1c1ccc(C)cc1C)OCC c1(C(=O)NC2CC(OC)C2)csc(CNC(=O)C(F)C2CCOC2)c1 C(=O)(C1(C)CCc2ccccc21)NCCC(CNC(c1c(OCC)scc1)=O)O C(=O)(C(C#N)C(C)(C)C)NC1C(NC(CCC2(C)CC2)=O)CCC1.C1C(=O)N1 C1(C(=O)NCCC2N(C(CC3CC(=C)C3)=O)CCC2)CC(OC)C(OC)C1 Cn1ncc([N+](=O)[O-])c1NCCCCCCNC(c1cccc(C(F)(F)F)n1)=O c1(C(C(=O)NC(CC)C)N(C)CCc2ccccc2)cc(OC)ncc1Br c1(OC)cnc(C(=O)NCC2CC(O)CN2C(C2CC2C(F)F)=O)nc1 c1(-c2cccc(C(C)O)c2)cccc2c1CN(C(=O)CS(=O)(=O)CCO)CC2 N1(C(c2c(CC)c[nH]n2)=O)CCC(C)(C)C1C(=O)NCc1ccoc1C N1(C(C(CC(N)=O)O)=O)CC(C2CCCN(C(c3nc[nH]c4nccc3-4)=O)C2)C1 C1(NC(c2ccc(C3CC3)s2)=O)CC2(C1)CC2C(=O)N(CCC1CCCS1)CCO CCC(CC1CCCC1)C(=O)NC1CC(CO)N(C(=O)CCc2cnn(C)c2)C1 c1(C(=O)NCC(CNC(C2C(COCC)C2)=O)(C)O)ncc(C)cc1OC N1(CC(=O)N(CC)CC)C2CCC1CC(NC(=O)C(=O)CC(C)C)C2 c1(C(N(C2CCCN(C(=O)C=CCF)CC2)C)=O)c[nH]c2ccc(Cl)cc2c1=O N1(C(c2cccc(N(C)C)n2)=O)CCCC2(C1)CN(C(=O)C(C)(C)CCC#N)C2 c1(CC)ccccc1NC(c1ccc(NC(=O)COC(C)=O)cn1)=O c1(CN2CCC(C)(C(=O)NCc3ccc(C=C)cc3)C2)c[nH]c2ncc(Cl)cc12 C1(NC(c2cc3c[nH]nc3s2)=O)CCOC2(CCN(C(C3CCCO3)=O)CC2)C1 C1(NC(C=NOC)=O)CN(C(c2ccc(=O)n(C)c2)=O)C2(CCOC2)C1 c1(OCC)cc(NC(C2(CNc3ncncc3C#N)CC2)=O)c(Br)cc1Br CC(CN(C)C)CC(=O)NC1(CCNC(c2cc(C3CC(F)(F)C3)[nH]n2)=O)CC1 C1(CNC(C(C)(C)CO)=O)N(C(=O)CCc2ccon2)CCCC1(C)C N1(C(CC2CC(CC)C2)=O)CC(C(=O)NCC2(C)CC2(C)C)CCC1(C)C c1(C(=O)NC(C)(C)CNC(c2cscc2Cl)=O)cnc2c(F)ccc(F)c2c1 n1(C(C)C)ccc(=NC(=O)CCNC(c2cc(C(N)=O)[nH]n2)=O)[nH]1 Cc1cc(C(=O)N(C2CCCN(C(=O)C(=O)N(C)C)CC2)C)nc(OC(C)C)n1 O=C(C1CCCc2nn[nH]c21)NCC(C1CCOC1)O C(=O)(C(CC(C)C)N(C)C(C1CC(O)CN1C)=O)N1C(C=C)CC1 c1(C(=O)NCCC)ccc(-c2csc(C(=O)NCc3sccc3Cl)c2)cc1 Cc1onc(CCO)c1C(N1CCC(C(C)NC(C2CC(C)(C)CO2)=O)CC1)=O c1(C(=O)Nc2nnc(C3(OC)CCOC3)s2)cncc2c1CCCC2 c1(C(=O)Nc2ncccc2O)c[nH]c2cc(-c3cc(C4CC4)cnc3F)cnc12 c1(C(=O)NC(C(=O)NCC#CC)Cc2cn[nH]c2)cccc(Cl)c1 C#CC1(OC(c2c(O)nnc(C)c2C)=O)CCC(C)(C)CC1 c1(C(N(C(C)CNC(c2ccc(CC(C)C)cc2)=O)CC)=O)ccnc(OC)n1 Cc1nccc(C(N2C(CNC(=O)C(C)C(C)C)CC3CC23)=O)c1O C(=O)(C1COCc2ccccc21)N1CCC(NC(c2cc(Cl)cc(Cl)c2)=O)C1 C(=O)(C(CO)C(F)(F)F)NC1C(NC(=O)OC(C)(C)C)COCC1 c1(C(=O)NCCCCNC(CC2(C)CCN(C(N)=O)C2)=O)cccc2ccnn12 c1(CC)ccc(C(N2CCC(C)(CC(=O)NC3CC(N(C)C)C3)C2)=O)nc1 C1(C(N2CC(=CC)C2)=O)CCCN(C(C2CN(C)CCO2)=O)CC1 c1(NC(C2C(C)(C)C(=O)C2)=O)cccc2n[nH]cc12 C=CC1CCCC(NC(C2COCCC2NC(C2(COC)CC(C)(C)C2)=O)=O)C1 c1(C(N2CCC(C(c3ccccc3)C)C2)C(=O)NCC=C)csc(C(C)C)n1 C1(C)(CNC(C(C)OC)=O)CC(F)(F)CN1C(c1ncc(C(N)=O)cc1Cl)=O C1(C(=O)NC2(CNC(c3c(N)cc(F)cn3)=O)CCOC2)CCOCC12CCC2 c1(CNc2ccc(C(=O)OC)c(O)c2)cc(F)c(Br)c(F)c1 CP(C)(=O)CCC(=O)NCC(CC1CCC(F)(F)CC1)CO C(C(CC(C)C)C(=O)N1CCN(C(=O)C=Cc2cccs2)CC1CC1CC1)OC c1(NC(C2CN(C(C3CC(O)C3)=O)CC2C(F)F)=O)nc(C2CC2)ncc1Cl C1(C(=O)NC2CC(C)(NC(c3cc(C(C)C)on3)=O)C2)CCOC(C)C1 c1(-c2nc(C)sc2)ccc(CC(=O)NCCCN2CCCC2C(=O)N(C)C)cc1 C#CCC(C)(CC)C(=O)NC1CCC2(CC1)CC2NC(c1coc(Cl)n1)=O c1(C2(C(=O)NC3(C)CC(NC(CCC=CC)=O)C3)CC2C(=O)O)cccc(Cl)c1 c1(C(=O)NCC=CCNC(C2CC2F)=O)cnc(C2CC2)[nH]1 c1(C(N2CCC(C)CC2)=O)cc2nccc(C(F)F)n2n1.c12sccc1NC2=O N1(C(c2cn(C(C)C)nn2)=O)CCC(C(=O)NCC2(C)CC3(CC3)C2)C(C)C1 C(=O)(CCC1=NNC(=O)CC1)NC1C(NC(C=Cc2cn(C)nn2)=O)CCCC1 c1(C(=O)NCCCN(CCCNC(C2C(=C)CC2)=O)C)cnc(Cl)s1 N1(C(C(CCN(C)C)O)=O)CCCN(C(C2(CO)CCCCC2)=O)CCC1 CN=c1ccc(C(=O)NC2CCC(CC(=O)NCCC(=O)NC(N)=O)C2)c[nH]1 c1(C(=O)NCC(CNC(C2=C(C)CCCC2)=O)O)c(Cl)cccc1[N+](=O)[O-] C#CC1COCCN1C(C1CCCN(C(c2c[nH]nc2Cl)=O)CC1)=O c1(CC(=O)NC23CC2CN(C(=O)CC2=CCCCC2)C3)ccc2c(c1)CCCC2 C(C(=O)N1CCOCC1c1cnn(C)c1)(C(C)C)SC N1(CC(=O)NCC2N(C(Cn3nnc(C)n3)=O)CC2)CCCCCC1=O C1(NC(C2CC(Cl)(Cl)C2)=O)CCC2(CCCN(C(=O)Cc3cncc(O)c3)C2)C1 C1(NC(C2N(S(CC)(=O)=O)CCC2)=O)CCC2CCC1N2 N1(C(C=Cc2ncc(C)[nH]2)=O)CC(NC(c2scnc2C)=O)CC2(CCC2)C1 c1(C(=O)NC(CC)CNC(c2ccc(F)nc2)=O)cn(C)c2c(cnn2C)c1=O C(=O)(CCCCO)NCC(N1CCC(C(C)(C)NC(c2cc(COC)n[nH]2)=O)C1)=O N1(C(C2C(C)(CC)C2)=O)CC(CNC(c2oc(SC)cc2C)=O)CC1C N1(Cc2cc(C#N)cn(C)c2=O)C2CCC1CC1(C2)CC1(F)F C(CCC(C)(C)C(=O)N(C1CCC1O)C)NC(CCCC1C(C)C1)=O CCCCC(C(=O)NC(C)C)N1CC(C(=O)OC)OC(C)C1 C(=O)(CS(=O)(=O)CC(C)C)NCC1CCN(C(c2c(C)ocn2)=O)C1(C)C C1(NC(CC2(C)CCC2)=O)CC(C2CCN(C(=O)CCOCCN(C)C)C2)C1 CN=c1[nH]c(=NCC2CN(CC(F)(F)F)C2)[nH]c(=NC2COc3c(F)cccc32)[nH]1 c1(CNC(=O)Nc2c(C(C)C)c(F)ccc2)cnc2ccnn2c1 N1(C(C2(N(C)C)CCOCC2)=O)CCN(C(c2cccs2)=O)C(C2CCC2)C1 c1(C(N)=O)cc(NC(c2cn(C3(C(F)F)CC3)nn2)=O)ccc1Br N1(C(c2ccc(C)cc2C)=O)CC(CNC(C2CCS2(=O)=O)=O)C2CCCCC12 C(CCN(CC(=O)NC)C(=O)C(F)(F)C(C)O)NC(CSCC=C)=O N1(C(CCc2nc(C)sc2)=O)CCCCC1C(C)NC(C1(c2cncs2)CC1)=O C1(C(=O)NCC2(O)CC(NC(c3cscn3)=O)C2)(CC)CCNC1=O C1(C)(C(=O)NC2CN(C(Cn3ncc(C#C)c3)=O)C3C2C3)CCN(C)CC1 C1(CNC(c2ccc(C(=O)OC)cn2)=O)CC2CCCC2N1C(=O)COCCF C1(CC=C)(NC(=O)CC(C)NC(N)=O)CN(C(C2(NC(C)=O)CCCC2)=O)C1 C12CCC=CC1NC2=O.C(=O)(CC(C)C1CC1)N1C(CC(=O)NC)CC1 c1(OC)ccccc1C(F)(F)C(=O)NCC1(NC(C2CC3CCCC23)=O)CC1 C1(NC(C2(CNC(c3ncc(C)c(C)c3)=O)CCC2)=O)CC2CC1CC21CC1 c1(C(N2CC(O)CC(NC(C=COCC)=O)C2)=O)cccc(S(C)=O)c1 C(CCC(N)=O)(C(=O)N1CC(F)CC1CN(C(=O)CC1CCC1)C)NC(C)=O C(=O)(CCCCCNC(=O)Cn1cnc(=N)[nH]1)NC(c1cccnc1)C CC1CN(C(=O)C(C)C(C)(F)F)CC1(C)CNC(C1(Cc2ccccc2)CC1)=O C1(COC)CN(C(=O)C(C)N(C(=O)CCC2CCCC2)C2CC2)CCO1 C(=O)(C1=CCC2(COC2)OC1)NC(C1CCN(C(C2(C)CCCC2O)=O)C1)(C)C c1(CCC)cc(C(=O)NC(C)CNC(C2CC2c2cccc(OC)c2)=O)sc1C CC1CN(c2cc(C(N)=O)ncn2)CCC1NC(=O)C(F)(F)c1ccnn1C C1(C(N(CC(CCC)O)C)=O)CN(C)CCN1C(c1cc(C)c(O)nn1)=O C1(CCNC(c2cccnc2S)=O)CN(C(=O)CC2CCC(F)(F)C2)CCCO1 C(=O)(C(CCC)NC(C1CCC1OCC)=O)NC(CC#CC)C CON(C)C1CN(C(=O)C(CNC(C2(CO)CC(C)(C)C2)=O)N(C)C)C1 CON(CCC(=O)N1CC(O)(C(C)C)C1)C(=O)C1(N(C)C)CCSC1 CCC(O)CC(=O)NCC1(C)CCN(C(=O)CN2C(=O)CNC2=O)C1 C1(NC(C(CC)CC)=O)CC(F)(F)CC1CNC(=O)COCCCC(C)C C(CCC(=O)NC(CNC(C1CC(C)(CC)C1)=O)C(C)C)OCCOCC N1(C(C(CNC(c2cc(C)on2)=O)C(C)C)=O)CC2CCC1C(O)C2O C12(C(N3CC(N(C)C(c4c[nH]c(=O)cn4)=O)C3)=O)CC1Cc1c[nH]nc12 Cc1cc(F)c(C(=O)Nc2c[nH]nc2Cl)c(Cl)c1 Cc1cc(O)cc(=O)n1C(C)C=O.c1(C)nnc2ncccn12 C1(CNC(=O)CCc2nncs2)CCCCN(C(C2CN3CCN2CC3)=O)C1 c1(C(=O)NCC(CC(C)C)NC(C(C)=C2CCC2)=O)cnc(O)c2ccsc12 N1(C(c2c(COC)noc2)=O)CCC(CNC(=O)C=CC2CCCCC2)CC1C c1(-c2n(C(C)C(F)(F)F)nc(-c3cnn(C)c3)n2)cccc2ccn(C)c12 C(=O)(N=c1cnn(C2CCOCC2)[nH]1)N1C(C)(C)CC1 CC12CC(NC(C3CC(=O)N(O)C3)=O)(C1)C1(CN(C(C3CCC(=O)N3)=O)C1)O2 c1(C(N2CCCC(CC)(NC(c3scnc3C)=O)C2)=O)cnn2c1OCC(O)C2 C1(NC(N(CC(c2ccccc2)CC)C)=O)CCN(CCOC)C1 C(CC(O)CC(=O)NCC1(C)CCN(C(=O)Cc2cnn(C)c2)C1)SC Cc1cc(CC(=O)NC2CC(NC(=O)C(C3CCC(=O)N3)C)C2)ccc1Cl N1(C(C2C(NC(CCC=C)=O)CCC2)=O)CCN(c2ccncc2)CC1 c1(OCC(=O)NCC=CCNC(C(C)N(C(C)=O)C)=O)cccc(O)c1 C=C1CCN(C(=O)CC(C)(F)F)C(C(=O)NCc2cnc(C)o2)C1 C1(CCOC)CN(C(=O)C(C)(C)C#N)CCN1C(=O)CC(C)(C)COC C#CCC(O)C(=O)NC(C1(O)CCCCC1)C(=O)OCC1COC1OC C(=O)(C1=CCS(=O)(=O)C1)NCCOCCCNC(=O)C#CC1CC1 c1(C(N2C3(CNC(C(C)(C)CO)=O)CCC3CC2)=O)ccc(S(N)(=O)=O)nc1 CCCC(C)CC(=O)N1CCOC(CC(N2CCCC(OC3CC3)C2)=O)C1 C1(C2CC2)(OC)CN(C(C23CC2CCN3C(c2cn(C)cc2C)=O)=O)C1 Cc1c(C(=O)NC2CCC(NC(=O)C(F)(F)C3CCCC3)CC2)cnn1CCO C1(NC(C=C(C)C2CC2)=O)CCN(C(C2CCCCS2)=O)C1 c1(C(C)(C)C)conc1CNCCCc1ccoc1 Cc1cnc(C(N2CC(NC(=O)CC3CCCCC3C)CC2C)=O)c(O)c1 C1(N(C(c2ccc(Br)o2)=O)CC)CCCN(C(c2ccnc(OC)c2)=O)C1 c1(C2C(C(N(C)CC3CCOC3)=O)C2)ccc(C(F)(F)F)cc1 C1(C(=O)NC(CC=CC(=O)NC(c2cc(C)on2)C)(C)C)CC(O)C(F)C1 N1(C(CCC#CC)=O)CCC2(CCN(C(=O)CCN3CCOC3=O)C2)C1 c1(OC)ccnc(CNC(=O)CCNC(=O)CCN2CCCC2=O)c1 N1(C(c2ccc(C)c(C#N)c2)=O)CCN2C(CCS2(=O)=O)C1 N1(C(CCc2c(C)noc2C)=O)CC(N(C(=O)COC(C)C)C)C2(CC2)C1 N1(C(C(CC(C)C)C)=O)CC2CCN(C(=O)C(C(C)C)C(C)C)CC2C1 n1(CC)cc([N+](=O)[O-])c(C(N2CCC(CO)C(NC(C3CCSCC3)=O)C2)=O)n1 Cc1cc(C(=O)NC(C)(C)C=CC(=O)N(C)CC2(O)CCC2)nc(C)n1 c1(C(N2C(CN(C)C(C3(C)CC4(CC4)C3)=O)CCC2)=O)ccc2c(c1)CCC2 CC1(C)CCC(CNC(c2coc3c2CCCC3)=O)N(C(=O)CCC#N)C1 CCC(CC(F)F)C(=O)N1CCC(C(C)C)CC1CNC(=O)CCCN(C)C CCCCCC(C)(C)C(=O)NCC(C)(C1CC1)NC(=O)CC1(C)CCS(=O)(=O)N1 C1(NC(CN2C(C)CCC2C)=O)CC2(C1)CN(C(=O)CN1CC=CC1)C2 c1(OC)ncc(C(=O)NC2CCN(C(c3cccc(C)c3O)=O)C2(C)C)c(C)n1 c1(C(=O)NCC(C)NC(C(C)OCc2ccc(C)cc2)=O)cccn2nccc12 Cc1cn2c(n1)CC(C(N1CC3CC1C3NC(=O)Cc1cncs1)=O)CC2 C1(C(CNC(CCOCCOCC)=O)NC(C2CCC2C)=O)CCCCC1 C12(CNC(Cc3c(C)cc(C)s3)=O)CCC1CN(C(=O)Cc1cccnc1Cl)C2 c1(C(=O)NC2CCC(NC(COC)=O)CC2)ccc(=O)n(CCO)c1 Cc1ccc2nc(C(=O)N(C3CC4CC3N(C(=O)C(C)C(F)(F)F)C4)C)cn2c1 CC1(C)CC(NC(c2csc(Br)n2)=O)CN(C(=O)CN=S(C)(C)=O)C1 N1(C(C(CCC2CCC2)NC(C2CCCCC2O)=O)=O)CC(C2CCCC2)C1 C#CC1CC2(CC(C(=O)NCC3(O)CN(C(=O)Cc4cccc(OC)c4)C3)C2)C1 C(CC(CC)C(=O)NCC1(NC(=O)CN2CCCCCC2)CCCCC1C)=CC N1(C(c2c(C)n(C)nc2)=O)CC2(CCN2C(=O)COCC2CCCCO2)C1 Cc1cc(O)c(Cl)cc1C(=O)NCC1CC(C)N(C(=O)COc2cc(C)on2)C1 c1(OC)cc(F)cnc1NC(=O)CC1(C)CN(Cc2ccncc2)C1 c1(OC)cc(Cl)c(Cl)cc1CNc1cccc(F)c1C(=O)Nc1ccc(SC)o1 Cc1ccn2cnc(C(N3CCOC(CCNC(c4cncs4)=O)C3)=O)c2c1 c12ncccc1-c1cccc(c1)SC2.c1(C(=O)NCCN2CCCC2)cscn1 c1(CN(CC(C)(C)NC(=O)Cc2n[nH]c(=N)s2)C)ccc(F)cc1 c1(C(=O)NCCN(C(=O)CO)CC)coc2c(Cl)cccc12 c1(C(=O)NCC2CCC(NC(CCS(C)(=O)=O)=O)C2)cnc(O)c2cccnc12 Cn1[nH]c(=N)cc1C(N1CC(CO)(NC(=O)C(c2ccccn2)O)C1)=O CCCCCCC(=O)N(C)CC1CCCN(C(=O)C(C(C)C)n2cc(C)cn2)C1 c1(N2CCCC(N(C(C(CCCC)C)=O)C)CC2)ncnc2sccc12 Cc1cnn(C)c1C(=O)NC(C)CN(C)C(c1cccc(C(C)C)c1)=O C(=O)(CCCCCNC(C1CC2(CCCO2)C1)=O)NCCCSC C1(NC(CCCCC)=O)CN(C(C2CC(=O)NC2(C)C)=O)C2(CCCCCC2)C1 c1(C(=O)NCC(O)CNC(C2CNc3ccnn3C2)=O)ccc2ccncc2c1 CC(c1ccco1)=CC(N1C(C(=O)NC2COC(C(C)C)C2)CCC1C1CC1)=O N1(C(c2cnc(C)n2C)=O)CC(C2CCCCN(C(=O)CCS(C)(=O)=O)C2)C1 Cc1ccc(C=CC(=O)NCC2CC2NC(=O)Cc2c(O)ncnc2O)nc1 CC(C)CC(C)CC(=O)N(C)CC1C2CN(C(=O)CO)CC12 S(=O)(=O)(CCC(=O)NCC(C(C)C(C)C)NC(=O)C=Cc1ncc(C)[nH]1)NC c1(C(C)C)nnc(N(CCCN(C2CCC2)C)C)n1Cc1ccccc1 C1(C(=O)NCCNC(CC)=O)CCCN(C(=O)CSCC(C)C)C1.C1CO1 C1(C(N2C(C)CN(C(=O)C(F)(F)c3ccccn3)CC2)=O)CC2(COC(=O)N2)C1 C1(C)(CNC(C(CCOC)C)=O)CC(F)(F)CN1C(=O)CC(O)c1ccccc1 N1(C(C(COC)(F)F)=O)CC2CCC(C1)N2C(C1(C#N)CCC1)=O C1(NC(c2cc[nH]n2)=O)CN(C(c2conc2C2CCC2)=O)CCC12CCC2 C(=O)(CCCCCF)NC(C(=O)NC1(COC)CN(C)C1)c1ccco1 c1(C2(C(=O)NCCCNC(=O)CO)CC2(Cl)Cl)ccc(Cl)cc1.C12CCC1N2 N1(CCC#C)CCC(C(=O)NCC2CCN2C(=O)CCN2CCCCC2=O)CC1 c1(C(=O)NCC(C)(C)NC(c2ccc(C(N(C)C)=O)[nH]2)=O)c(C(N)=O)cnn1C N#CCS(=O)(=O)c1ccc(C(=O)Nc2cnc(C3CCNCC3)nc2)cc1 Cc1scc(C(=O)NCCC2(C)CCN(C(=O)CCc3ncccn3)C2)c1C C1(CN(C(=O)CCCOC(C)C)CC)CCN(C(=O)C(C)Cn2cccn2)CC1 c1(CNC(CC(CC)N(C)C(C2(C)CCN(C)C2=O)=O)=O)cc(C)cnc1F S(=O)(=O)(c1cn(C)cn1)N(C)CCC1CCOCC1 C1(C(=O)NC2CC(CNC(C3(S(N)(=O)=O)CC3)=O)CC2O)CCc2cnnn2C1 C(=O)(C1CCc2c[nH]nc21)N1CCN(CC(=O)NCC(C)CN=[N+]=[N-])CC1 C(CC(C)C)(C(=O)NCC1(C(C)NC(=O)COC(F)F)CC1)NC(C)=O c1(NC(C2C(CCC)CN(C(=O)C(CC3CC3)OC)C2)=O)ccc(F)c(F)c1 C1(C(N2CC(O)(CNC(Cc3cc(C)on3)=O)C2)=O)COC(=O)N1C C=CCCCCCCC(=O)NCCC1(C)CCN(C(c2cnc(C)s2)=O)C1 C1(CCCC(=O)OC)CCN(C(=O)Nc2cncc(C3CC3)c2)CC1 C1(C#N)(C(=O)NCC(C(C)(C)C)NC(=O)Cn2ncccc2=O)CC(F)(F)C1 C(C(C)(C)C(=O)NC1CC(C(F)F)C1)NC(C(C)NC=O)=O C(=O)(C(C#N)C(C)(C)C)NC1C(C(=O)NCc2cc(C)c(C)s2)CCC=C1 N1(C(c2cc(C)c(C)o2)=O)CCCC(C)(C)C1C(=O)NC1CCCC1 N1(C(c2ccc3ncoc3c2)=O)CCC2(CCN(C(c3cnco3)=O)C2)C1 Cc1cc(C(N2CC3(CC3C(=O)Nc3ccc(F)c(Br)c3)C2)=O)ccc1Br N1(C(c2ccc(C)n2C)=O)CC23CCCC2(C1)CN(c1nc(C#N)c(Cl)s1)C3 c1(C(N2C(CNC(c3[nH]c(C)cc3C)=O)CC(OC)C2)=O)[nH]nc([N+](=O)[O-])c1Cl C1(C(=O)NCC2OCCO2)(OC)CCN(C(=O)CCC2CCC(O)CC2)CC1 C1(C(N2CCCC(CNC(=O)CC3CCCCCCC3)C2)=O)CCCCNC1=O n1(CC(=O)NC2CC3(CCN(C(C4CCCC5CC45)=O)C3)C2)cc2ccccc2n1 c1(OC)cc(-c2ccc(F)cc2C(=O)O)c2c(c1)CCO2 CN1CC(C(=O)NCc2cc(C(N3CCC(CF)C3)=O)no2)CC1=O c1(C(=O)NCCn2c(C)nnc2)cncc2nc(O)[nH]c12 N1(C(CC(C)(O)C2CC2)=O)CCCCC(NC(=O)COC2CCCC2)C1 C1(C(N2CCC(CCCC)C2)=O)CN(C)CCN1C(C1CC(=O)C1(C)C)=O C12(CNC(=O)C#CC3CC3)CCC1CCN2C(=O)CCc1nc(C2CC2)no1 N1(Cc2ncn(C)c2)CC2C(C(N3CCCC(CCCO)C3)=O)C2C1 Cc1cc(F)ncc1NC(C1CN(C(c2ncnc(C)c2C)=O)CC1(F)F)=O N1(C(C(C)C#N)=O)CCC(CN(C(c2cccc(=O)o2)=O)C2CC2)CC1 C(CNC(=O)C(c1cccs1)NC(=O)Cn1cc(CO)nn1)(C(C)(C)C)OC c1(C(N(CCCN(C(C2C(C=C)C2)=O)C)C)=O)sc2nccn2c1C c1(C(C(=O)N(CC(C)NC(c2cc(Br)c[nH]2)=O)CC)C)ccncc1C C=CCCCCCC(=O)NC(CCN(C)C)C(=O)N(C1CCOC(C)(C)C1)C C1(C(=O)NCC2N(C(c3cncc(C(=O)OC)c3)=O)CC2)CCCC(C)(C)O1 C(CC(C)C)(C(=O)NCCCN(C)C(c1cc(C2CC2)ncn1)=O)NC(C)=O Cc1cc(C(=O)NC2CCCC2NC(=O)C(C)(C)c2ccns2)c(C)o1 C1(CC)C(=O)N(C)CCN1C(C1(N)CC(CO)C1)=O.C(=O)(C(C)OC(C)=O)C(C)=O c1(-c2ccc(C#N)o2)csc(=Nc2ccc3c(c2)OCCCO3)n1CC1(F)CC1 C(=O)(C1CSc2ccccc21)NCC1CC(OC)CN1C(=O)CN(C)C(C)C C12(CNC(c3c(C(C)C)ncs3)=O)CC(NC(=O)CCCCN(C)C)(CO1)C2 CCC(COC)(CC)C(=O)N(C(C)CC(=O)NCC(C)(F)C(C)(C)F)C S(=O)(=O)(c1c(F)c(F)cc(F)c1F)N1CCOCC(CN)C1 N1(C(C2CCC(CC)CC2)=O)CCN(C(c2cnsc2C)=O)C(CC2CC2)C1 Cc1occc(=O)c1OCCn1cc(C2CCN(C(=O)CC3CC3)C(C)C2)nn1 C1(C(=O)NCC(CCOC)NC(C2(C)CC(C)C2)=O)CCn2c(O)nnc2C1 C1(CCC(=O)NCCCN(C(=O)C=Cc2ncc[nH]2)C)CCCC(O)C1 Cc1cn2cc(C(N3CCC(N(C(=O)COCP(C)(C)=O)CCO)CC3)=O)nc2s1 N1(C(C(N2C(=O)CCC2=O)C)=O)CCC2(C1)CN(C(=O)COc1ccc(O)cc1)C2 c1(CN=C(NCC2CCN(C)CC2)NC2CCCCC2)nnc2n1CCOC2 C1(C(=O)NCCCC(C)NC(=O)C(C)Cc2ccccc2)CCN2CCOCC12 c1(C(N2CCC(CNC(C3(CC)CCOC3)=O)C2)=O)ccc2[nH]nc(O)c2c1 N1(C(CCCOCCOC)=O)CC2CC(NC(=O)CCOC3CC3)C1C2 N1(C(C(CC(C)C)C)=O)CC(C)CN(C(c2cnc(O)n2C)=O)CC1C N1(C(c2nc(C(C)C)sc2)=O)CCC(F)(F)C(CNC(c2snc(Cl)c2Cl)=O)C1 N1(C(C2CCC(C)NC2=O)=O)CCN(C(=O)CCCS(C)(=O)=O)C2(CCC2)C1 Cc1cc(C)n(-c2ccnc(NC3CC(NC(=O)Cn4nccn4)C3)n2)n1 c1(C(N2C(C)C(C(=O)NCCC(Cl)Cl)CC2)=O)ncn2c1CCC2 CC(C(=O)N1CCC(CO)(NC(=O)C=Cc2ccc(C(F)F)o2)C1)C(F)F C1(F)(CNC(Cc2cc(C)ns2)=O)CCCN(C(c2ncccc2N)=O)C1 N1(C(c2cc(OC)c(C)cc2)=O)CC(C2CCCN(C(=O)C(F)(F)C(C)O)C2)C1 Cn1nccc1C(=O)NC(CO)C(=O)NCC1C2CCCC12 CC(C)(O)C(=O)NNC(=O)c1cccc(S(=O)(=O)N2CCC(N)CC2)c1 N1(C(c2c(OC(C)C)ccc(OC)c2)=O)CCN(C(=O)CNC(C)=O)C(CO)C1 N1(C(c2c(C)nc[nH]2)=O)CCC12CN(C(C1OCCC1c1cnn(C)c1)=O)C2 C1(NC(CCN(C(CCC)C)C)=O)COCCN(C(c2ccc(N)cn2)=O)C1 c1(C(N2C(CNC(C(c3scc(C)n3)C)=O)CC(O)C2)=O)cncc2nc[nH]c12 c1(CC(=O)NCC2CC(O)CN2C(C2CC3CCC3C2)=O)cnc2cccnn12 N1(C(C2N(C)CCOC2)=O)CC2(CCC(CNC(C34COC(CCO3)C4)=O)O2)C1 CC1CCCN(C(c2coc3c2COC3)=O)C1CNC(c1ccc(CF)cc1)=O CC(C)CCCCCC(=O)NC1(C2CCN(C(=O)C3=CCCC3C)C2)CC1 Cc1cn(C(C)(C)C(=O)N2CCC(NC(C3CCOC3)=O)C2)cn1 n1(CC(C)NC(=O)CC(=O)N(C)C)cc(CC2(O)CC(C(=O)OC)C2)nn1 C1(NC(c2c(C)onc2)=O)CC(NC(=O)C(N2CCSCC2)C)C(O)C1 C1(NC(c2nc(CCCC)sc2)=O)CCN(C(c2coc(C)c2)=O)C12CCC2 C1(C(N(CCNC(=O)OCCO)CCOCCO)=O)CC2CC12 C1(C(N(C(C)CCNC(C2(NC(=O)OC(C)(C)C)CC2)=O)C)=O)CC#CCCO1 C1(CCNC(C2CCCCS2(=O)=O)=O)CCN(C(c2cncs2)=O)CC1(F)F C1(c2nnnn2C(C)C)(NCc2ccc(C)c(C(F)(F)F)c2)CCN(C)C(C)C1 c1(N(C(=O)Cc2nc(Cc3cc(O)no3)no2)CC)ccc(F)cc1 c1(C(=O)NCC2CC3CN(C(c4ncc(C)nc4)=O)CC32)nccc(C#N)c1F c1(COC)nc(NCc2cc(C)cnc2O)cc(=NCCN2CCSCC2)[nH]1 c1(C(=O)NCC2C(NC(=O)CCCc3nccs3)C2)cc2ccc(F)cc2cn1 N1(C(C(CC2CC2)NC(C(C(C)C)C#N)=O)=O)CCC12CCOCC2 N1(C(c2ccc(C)s2)=O)CCC2(CC1)COC(CNC(C1CC(C#N)C1)=O)C2 C1(C(=O)NC2(COC)CCCC2)CCOCC1NC(=O)C1CC1 c1(C(=O)NCCN(C(c2c(O)cc(C)nn2)=O)C2CC2)ccc(C)c(C)c1Cl CC(C)C(C(=O)NC1CC(F)(CNC(=O)CC2CC2(Cl)Cl)C1)NC(N)=O CC(C)CC(O)C(=O)N1CCCC1CNC(=O)Cc1sccc1-c1ccccc1 C1(CC(=O)NCC(CC)NC(c2snnc2C(C)C)=O)CCCC(OC)C1 C(=O)(C(CCOCCO)NC(=O)CN(C1CCCC1)C)N1CC(O)(CC=C)C1 c1(N(C)C)ncc(CNCC2COCC2N(C)C)s1 N1(C(c2cc(C)oc2C)=O)CC(C)C(NC(=O)CCc2ccsc2Cl)C(C)C1 Cc1nnn(C)c1-c1cccc(CC(=O)N(C)C)c1 C1(N(C(=O)CCc2cnoc2)CC)CCCN(C(=O)C(COC)CC)C1 N1(CC2(CO)CCOC2)CCCOCC1.c12cn(nn1)C2 Cc1ccc(F)c(C(=O)NC(CN(C)C)C(=O)NC2C3CCCCCC23)c1 c1(C(=O)OC)coc(C=CC(N2CC(NC(=O)CC3CCC4CC34)CC2C)=O)c1 Cc1c(C(=O)NC2(CO)CCN(C(=O)C(C)Oc3cccnc3)C2)cccc1O N1(C(C(=O)NCC)=O)CCC2CCCC12C(=O)NCc1cncc(C)c1 c1(CN(C(C=CC(C)NC(=O)CO)=O)CC2CCCC2)cc(=O)cc[nH]1 Cc1cc(CN2CCOC(CNC(c3cnc(Cl)cc3I)=O)C2)c(F)cc1Br C(C(C(=O)N1CCN(C2CN(C(=O)C(F)OC(F)(F)F)C2)CC1)C(F)(F)F)OC N1(C(c2c(C)cno2)=O)CCCCCC(NC(C2OCC3COCCC23)=O)C1 N1(C(c2c(COC)noc2)=O)CCC2(NC(c3nn(C)c(C)c3Cl)=O)CC2C1 C1(C)(C(=O)NC(CNC(C(C)NC(=O)Cn2cnnn2)=O)(C)C)OCCO1 c1(CC)nccc(N(CC(C)CNC(=O)Cc2cc(C)no2)C)n1 C1(C(=O)OCCC(C)(C)O)CC(NC(=O)CN2CCC(O)CC2)C12CCC2 c1(C(N(CCN(C(=O)C(C)C2CCOC2)CC)CC)=O)cnoc1C1CCC1 c1(-c2cc(C(=O)NC3C(NC(c4n(CC)ncc4)=O)C3)no2)ccc(Cl)cc1Cl C1(C(N2CCC(C=C)C2)=O)COC2(C1)CN(C(=O)C#CC1CC1)C2 N1(C(CC=C)=O)CCN(C(c2c(C)cc(C#N)cc2C)=O)CC12CCC2 c1(OC)ncc(C2=CCC(C)CC2)cc1C(=O)N(CC(F)(F)F)CCN c1(C(=O)OCC)cc(C)c(NC(=O)NCC2CC(n3cccn3)C2)cc1F C1(C(=O)NC2(CC)CCCC2)CN(C(=O)C(=O)NOC)C2(CCC2)C1 CCCCC(O)C(C)C(=O)N1CC(NC(C2CS(=O)(=O)C2)=O)CC1C C1(C(C)NCC(=O)Nc2ccc(OCC3CCCO3)nc2)CN(CC)CC1(C)C C1(NC(Cc2c(C)n(C)nc2)=O)COCCN(C(c2nc(O)[nH]c(=O)n2)=O)C1 N1(c2[nH]c(=NCc3n(CC)c(C)nc3)[nH]c(=N)n2)CCC2(CCCNC2=O)CC1 CCCCC(=O)N(C)CCN(C(C1CCCO1)=O)C(C)C N1(C(C(C)NC(C)=O)=O)CC2CCN(C(c3ccc4n[nH]cc4n3)=O)C2C1 c1(C(N2CC(C)C(NC(C3CCCC4(CC4)C3)=O)C2)=O)cc(Cl)ccc1Cl c1(C(=O)NCCCNC(C(CSC)OC)=O)cn(C)nc1C c1(C(N(C2CC(C(N3CCCC4CC34)=O)C2)C)=O)cc(F)ccc1F N1(C(C2(OC)CCCC2)=O)CC(NC(=O)CN2CCCC(N(C)C)C2)C(SC)C1 c1(C(CNC(=O)COC(C)(C)C)NC(C2C(OCC)CC2)=O)cccnc1 c1(C(C(=O)NCC(COC)O)NC(c2cnsn2)=O)cn(C)nn1 N1(C(C(C=CCCC)O)=O)CC(CNC(=O)CCC(=O)N(C)C)C2(CC2)C1 c1(-c2cn(CC3N(C(c4ncn(C)c(=O)c4)=O)CC3)nn2)cnc2cccnn12 c1(C2C(C(=O)NCCCNC(C3CCCC3O)=O)C2)cccc(Cl)c1Cl C12(NC(C(c3ccccc3F)C)=O)CCOC(CNC(=O)C(O)P(C)(C)=O)(C1)C2 C1(F)(C(N(CCCCN(C(=O)C(F)n2ccnc2)C)C)=O)CC=CCC1 N1(C(=O)CC=Cc2cccc(F)c2)CCOCc2cc(Br)ccc21 C1(C(=O)NCCCN(C(c2cccc(C(F)F)c2)=O)CC)CCCC(N(C)C)C1 C1(CSC)CCC(NC(C2(n3cc(-c4nccc(C)n4)nn3)CC2)=O)CC1 C(=O)(CC(COC(N1CC(n2cccc2)C1)=O)OCC)OC.C(C)(C)(C)OC=O c1(C(=O)NC(CC)CNC(=O)C(F)(F)c2cncs2)cnc2ccnn2c1C c1(C(N(CC(CNC(c2c(COC)nn[nH]2)=O)O)C)=O)cnccc1N(C)C C(=O)(C(C)(C1(C)CC1)OC)N(CC(=O)NCCOC(CC)CC)CC#C C1(CNC(c2nc(CS(C)(=O)=O)sc2)=O)CC2(CCC2)CN1C(=O)C1=CCCC1 c1(C(N(CCOCCCNC(C(CC=C)(F)F)=O)C)=O)[nH]nc([N+](=O)[O-])c1Cl c1(CC(C(=O)O)NC(C(C)NS(CC)(=O)=O)=O)ccc(OCC)c(F)c1 c1(NC(C(=O)NC(CC#CCCCNC(C)=O)C2CC2)=O)cc(S(N)(=O)=O)co1 C(=O)(C(C(C)NC(c1ccnn1CCF)=O)C(C)C)Nc1cccc(COC)c1 C(=O)(C(N=[N+]=[N-])C(C)C)NC(COC)C(N1CC2(CNC(=O)C2)C1)=O C(=O)(CC(=O)OC)N1CC(C(C(=O)N(CC(CC)OC(C)C)C)O)C1 CN1CCC(NC(=O)C=CCN(C(=O)COC2CCCCC2)C)C(C)(C)C1 C12(NC(C3CCN(C)C3)=O)CCCC1N(C(=O)CCc1ccc(Cl)cc1)CCC2 CC(CCCCO)NC(=O)CC1COCCN1C(=O)CCCC1CC1C CN1CC2(CCN(C(c3cc(CNC(c4c(C#N)ncn4C)=O)[nH]n3)=O)CC2)C1 c1(C(=O)NC(C2CN(C(c3ccn(CC)n3)=O)C2)C)c2n(c(=O)n1C)CCCC2 C1(C(N2C(C(=O)NC(c3ccncc3)C)C=CC2)=O)CC12CCCCC2 N1(C(C2C(C)C(=O)C2)=O)CC2(CCC(CNC(C3C(C)(C)C3(F)F)=O)O2)C1 N1(c2cc(C)[nH]n2)CCN(C(c2cncn2C(C)C)=O)CC1 C12(NC(C(c3cc(C)sc3)(C)C)=O)CCCC1CN(C(=O)Cc1csnc1C)C2 c1(OC)ccncc1C(=O)NCCCC(C)NC(C1CC(C(C)(C)C)C1)=O C1(C(N(CC(=O)NC2(COC)CC2)CC2CC2C)=O)CC2OC1C1CC21 C1(CC(N)=O)CCCN(CC2CC(=O)N(c3cccc(Cl)c3)C2)CC1 c1(CC)nn(C)cc1CNC(=O)C(CN(C)C)NC(=O)Cc1cc[nH]c1 C(=O)(C(C#N)CC1CC1)NC(C(C)NC(c1c(CC)ocn1)=O)C CCS(=O)(=O)CC(=O)NCC1CC2(CC2)CN1C(c1scnc1C1CC1)=O c1(CC)nccnc1C(=O)NCC1(F)CN(C(C2CN(C)CCO2)=O)C1 Cc1coc(C)c1C=CC(=O)NC1CN(C(=O)C(c2cnn(C)c2)C)CC1C c1(CCC)cc(C(N2CCC(N(C)C(C3(C)CC3(F)Cl)=O)CC2)=O)ccn1 C=CCCCCCCC(=O)N1CCC(CNC(=O)CCCC#N)CC1C N1(C(=O)C=C2CCOCC2)CC(C(N2CCC(C(F)(F)F)C2)=O)C(F)(F)C1 C=CC(C)(CC)C(=O)NC(C1CN(CCn2cc(Cl)cn2)C1)C CCCCCC(C)CC(=O)N1CCC(C)C(CNC(=O)CCc2cc(C)no2)C1 N1(C(CNC(CCC)=O)=O)CCN(C(c2cnn(C3CCC3)c2)=O)CC1C1CC1 C(CCN(C)C(c1cc(C2CCOCC2)on1)=O)(C(C)C)NC(COCC#C)=O C(=O)(C#Cc1ccccc1Cl)N1CCC(N(CCCCCC)C)CC1 Cc1[nH]nc(C(F)(F)F)c1C(=O)NCC(C1CCC1)NC(c1cnn(C)c1F)=O CC1CN(C(=O)C(CO)NC(N)=O)CCN1C(=O)CC(C)(C)N(C)C C(=O)(CCC(=O)NCc1ccc(NC(C2CCN(C)O2)=O)nc1)NCCC c1(C(=O)OC)oc(C(=O)NCCC(C)NC(=O)CSc2ccc(F)cc2)cc1C c1(CC)cnc(O)c(C(=O)NCCC(C)NC(c2cc3scnc3[nH]2)=O)c1 C(c1ccc(C(C)C)cc1)=CC(=O)NC(CNC(C(C)(C1CC1)OC)=O)C(C)C c1(NC(C(C)OCC(C)C)=O)ccc(NC(=O)CC2CCCCO2)nc1 Cc1ccc(C(=O)NCC(C)(O)CNC(c2cc(F)n(C)n2)=O)c(N)c1F C1(C(N2CC3C(C(N(CC(C)O)CCF)=O)C3C2)=O)CC2CCCC2C1 C(C(C(=O)N(CCO)CCO)NC(c1cc(OC)ns1)=O)OCC c1(C(N(C2CCCN(C(c3cc(Cl)cnc3O)=O)C2)C)=O)ccc(Br)c(Cl)c1F C(=O)(C1=NOC(CNC(=O)CC2CSCCO2)C1)N1CCN(CC#CC)CC1 C1(C2(N)CCC2)(C(=O)NCc2ccc(C(C)C)cc2)CCC1 C(C(=O)N1CCC1CNC(=O)C(C)(C)n1cnnn1)(C(C)(C)C)OC c1(C(N2C3CC(NC(C(C)n4cccn4)=O)C2CC3)=O)c[nH]c2nccc(Cl)c12 c1(C(N2CC(C(N3CC(C(N)=O)OCC3)=O)C(O)CC2)=O)cn2ccsc2n1 c1(C(=O)NC(CN(C(=O)C(F)CC2CCC2)C)(C)C)cc(-c2ccncc2)on1 c1(C(N(C2CC(NC(C(COCC)C)=O)C2)C)=O)ccc(F)c(CC)c1 C1(C(=O)NC(C)CN(C)C(C2CC(F)(CF)C2)=O)CCc2nc[nH]c2C1 c1(CN2CCCC(C(C)NC(=O)CN(C)CCN(C)C)C2)ccc(C#N)cc1 c1(C(=O)NCC2(F)CCC(NC(C3CCN(C(N)=O)C3)=O)C2)cc2cnccc2o1 N1(C(CCC2C(C)C2)=O)CC2CC1CN2C(=O)CN1CCC(F)(F)C1 C#Cc1cccc(CNC(=O)C(CC2CCCC2)NC(c2cnnn2C=C)=O)c1 C#CC1(C(N2CC(S(C)(=N)=O)C2)=O)CCN(C(=O)CC2(O)CCCC2)C1 N1(C(c2c(OC)noc2C)=O)CCC(CNC(=O)C(C)(O)C2CCC2)C12CCC2 c1(C(N(C2CCN(C(=O)C3=CC(C)(C)C3)C2)C)=O)ccc(Cl)c2cccnc12 c1(C(N2C(CNC(C(CO)N(C)C)=O)C=CC2)=O)cc(Cl)c(Cl)cc1N CC(CNC(=O)Cc1ccnc(O)c1)CC(=O)NC1CCN(C(C)(C)C)C1 N1(C(C2CN(C(Cc3ccc(C)o3)=O)CC2C(C)C)=O)CC2(CCC2)C12CCC2 C1(CCNC(=O)C=CCO)CCCN(C(=O)CCC(=O)c2cccs2)CC1 N1(C(C(CC#C)C)=O)CCC2CCN(C(c3nccc4[nH]ccc34)=O)CC12 CCC(C)(C)C(O)C(=O)N1CC2(CC(CC(N3CC4CCC3C(CO)C4)=O)C2)C1 CC(C)C(CNC(=O)C1=CCN(C)C1)C(=O)NCC(O)CF CCC(O)C(F)(F)C(=O)N1CCN(C(c2ncnc3[nH]ccc23)=O)CC1C O=C(C1=CCCN(C(=O)CCC2OCCO2)C1)NC1(CCN2CCCC2)CCC1 c1(C(=O)NC(CC)(C)CNC(c2cc(OC)no2)=O)cnn2ncccc12 S1(=O)(=O)c2cnc(s2)Nc2c(scc2)C(=O)N1C(c1csc(C)n1)=O.CCOC c1(OC)cc(F)c(F)cc1C(=O)NCC(O)CNC(c1nn[nH]c1Cl)=O CC1CCN(C(=O)CCC2NC(=O)NC2=O)CC1NC(c1cncc(Cl)c1Cl)=O N1(C(c2cc(CCNC(c3c(C)ccc(F)c3)=O)on2)=O)CCC2(C1)CC2(F)F N1(C(CC2C(C)CCCC2)=O)CC2CCCC(NC(C3(C)CNC(=O)C3)=O)C2C1 Cc1cc2n(n1)CCN(c1ncccc1S(=O)(=O)NC1CCCCCC1CO)C2 c1(C(N2C(C(C)(C)NC(CCOCCOC)=O)CCC2)=O)ccc(F)c(Cl)c1F CN1CCCC1=NS(=O)(=O)c1ccc(NC(=O)NC2OC3CCC2CC3)cc1 c1(C(=O)NCCCN(C)C(c2ccccc2Br)=O)ncccc1Cl CS(=O)(=O)c1csc(CNCc2cscc2C(=O)O)c1 Cc1nc2c(cc1C(=O)OCC1CC3(CC3)C1)CCCN2C(=O)OC(C)(C)C CC#CCCCC(=O)NCC(O)CCNC(=O)C=Cc1ccc(C)o1 c1(SCCC(=O)N(CC(C)C)Cc2ncc(C)s2)ccc2c(c1)OCCO2 C12(CNC(c3nn(CC)nc3Br)=O)CCCC(CN1C(=O)C(C)CS(C)(=O)=O)C2 Cc1ccc(F)cc1C(N1CCCC1CN(C(=O)CC1COCC1O)C1CC1)=O N1(C(CC(C)OC)=O)CCC(CCNC(=O)C=Cc2ncco2)C(F)(F)CC1 c1(C(C(=O)NC2CC(NC(CC=C(C)C)=O)C2)C)ccc(F)cc1 N1(C(CC(C)Nc2cncn2-c2ccccc2)=O)CCN(CC)CC1C C1(NC(c2ncc(OC)cc2F)=O)CN(C(=O)CC(C)P(C)(C)=O)CC12CCC2 C.C1(=O)CNCCN1CCN(C(COCCOC)=O)C.C(C)(C)S c1(NC(C2C(NCc3ccc(CC)o3)C2)=O)ccc2n[nH]cc2c1C C1(CC(=O)NCC(CC)NC(C2CCCOC2)=O)CCCCC1(C)C C1(C)(CNC(C=CC(C)(C)NC(CCc2n(C)ccc2)=O)=O)CC2CC2C1 C1(OC)CC(NC(=O)CCCCn2ccnn2)CN(C(c2ccn(C)n2)=O)C1 C1(NC(C2(OCC)CCC2)=O)CCCC1CNC(C1CCN(CC(F)(F)F)C1)=O C12(C(=O)NCC(C(C)C)NC(c3c(C)cccc3N)=O)CCC(CC1)C2(C)C N1(C(CNS(CC)(=O)=O)=O)CCN(C(c2sc(N(C)C)nc2Cl)=O)CCC1C CC1(C)CCC(C(=O)N(CCNC(=O)CC(F)F)Cc2ccccc2)CO1 C1(NC(CSCC#C)=O)CCN(C(c2cc(CC)ccn2)=O)CC1C(C)C C(N=c1nc(N2CCOCC(C)C2)c2ncn(CC)c2[nH]1)C1(CCOC)CC1 Cc1nc(NCC2CCCCC2NC(=O)Nc2oncc2C)cc(O)n1 N1(C(c2cc(C)nc(Cl)c2N)=O)CCCC2C1CCCN2C(c1csc(Cl)c1)=O C=CC(C(=O)NCC(C)CNC(c1ccc[nH]1)=O)c1ccccc1 N1(C(c2c(C#N)scc2)=O)CC(C(N2CC3OCCOC3C2)=O)C(C2CC2)C1 N1(C(C2(SC)CC2)=O)CCC2(CCC(NC(=O)CC3CC(F)(F)C3)C2)CC1 C1(CN(CCOC)C)CCCCN1C(c1cccnc1)=O c1(C(CSCC2C(OC)(OC)CC2)=O)c(N)c(C(F)(F)F)nn1C.C(C)=O CC1=CCC(C)(C(=O)NC2CC3CC2N(C(c2cccc(C(F)F)c2)=O)C3)CC1 C1(OC)CCN(CC(c2c(F)cccc2F)C)CC1C C1(CNC(=O)Cc2ccno2)CCCN(C(=O)C=CC2CCCC2)C1 C1(NC(c2c(C(C)(C)C)nc(C)s2)=O)CCCCN(C(c2cocn2)=O)CC1 c1(CC)cc(C(=O)NC(C)CC(C)NC(c2ncccc2C(C)(C)C)=O)c(C)o1 N1(C(COCCCOC)=O)CCC2C(C1)CN2C(=O)CCc1cccn1C N(C(=NCCCCC(C)(C)C)NCCF)C(C)CCC(=O)N(C)C C1(C)(C(N2CC(NC(CC=CC)=O)C(C(F)(F)F)C2)=O)CCC(C)CC1 C1(NC23CCC(CNC(=O)OC(C)(C)C)(OC2)C3)CCc2nnnn2C1 C(C)(C)(CC(F)C(=O)NCCc1cc(C)ns1)NC(C(CCCC)F)=O N1(C(C(C)CNC(=O)CCc2ccnn2C)=O)CC(C)CC(C)(C)C1 C1(OC(CC)=O)CCN(C(=O)CCC2(C)CN(C(c3cc(OC)cs3)=O)C2)C1 Cc1ccc(NC(C2OCCC2CNC(c2nnc(S)n2C)=O)=O)cc1F C1(CC)(CNC(=O)NCc2ccccc2C(=O)O)CCOCC1 C1(C(=O)NCC(C(=O)OC)C)(CNC(=O)C=C2CCC2)CC12CCC2 c1(CCCC)ccc2nc(C(=O)N(C(c3ccccc3Br)C(=O)O)C)oc2c1 N1(CCC)CCCCC1C(=O)NC1CN(C(=O)Cc2nnc(C)s2)CC1C(F)F c1(C(N(CC(CN(C(C(CC)NC(C)=O)=O)C)O)C)=O)ccn(C2CC2)c1C c1(NC(CC2C(C)=NN(c3ccccc3)C2=O)=O)nc2c(s1)C(=O)NCC2 C=CCC(CNC(C1CCNC1=O)=O)C(=O)Nc1cn(C)nc1OC N1(C(C2(C)C(C)CCC2)=O)CCCC(C2CC2NC(=O)C2Cc3ccccc32)C1 c1(C(=O)NCC(CNC(C(C)NS(CC)(=O)=O)=O)(C)O)cc(O)nc(O)c1 N1(C(c2cc(SC)cc(Cl)c2)=O)CC2CN(C(C3CNC(=O)C3)=O)CC2C1 C=C(C)CCCC(=O)NC1C2CC1N(C(=O)CC1=CCCC1)C2C c1(C(=O)NCC2(O)CN(C(C(CCSC)OC)=O)C2)cc2ccccc2c(=O)o1 C1(C2CN(C(C3CCS3(=O)=O)=O)C2)(NC(=O)CCc2cccnc2)CC1 CCCC(O)C(=O)NCC(CNC(c1cn(C2CNC2)nn1)=O)CO C1(C(=O)NC2COCCN(C(C3(CF)COC3)=O)C2)CCC2(CCOCC2)O1 N1(CC)C(C)CN(c2nc(C)nc(-c3ccccn3)c2C)CC1C C(C)(C(=O)NCCOCC1CCN(C(c2c[nH]nc2C)=O)C1)(C1CC1)OC c1(C(=O)NCC(C)CNC(c2cn(C)nn2)=O)nn[nH]c1C(F)(F)F C1(N(C(C(N)=O)CO)C(=O)Cc2ccccc2O)CCCC12CCNCC2 C12(C(=O)NC3C(C(=O)NC4(CC)CCCCC4)COCC3)CCC(C1)OC2C N1(C(CCCOC(C)C)=O)CC(CNC(=O)CCCN(C)C(C)=O)C2CC12 c1(COC)cccc(C(=O)NCCOCCCNC(C2CCC(F)C2)=O)c1 C1(NC(c2ncc(CC)cn2)=O)CCCCN(C(=O)C(C)Oc2ccccc2)C1 C(N=C(NCC1CCCO1)N1CCC(O)CC(C)(C)C1)c1nc(C)cc(NC)n1 c1(C(=O)NCC2N(C(c3c(SCC#N)cccc3)=O)CC2)cc2c(s1)CCSC2 CC1CCN(C(=O)C#CC(C)(C)O)CC1C(=O)N(C)C.C1(=O)CCCN1 C(=O)(C(F)CC(C)C)N1CC(O)(C(CNC(CCc2onc(CC)n2)=O)(C)C)C1 CN(C)NC(=O)CCC(=O)NC1(C(=O)N(C2CCC2)C)CCCC1 C#CCC(O)C(=O)NC(c1ccccc1F)CNC(c1ccoc1C1CC1)=O C(=O)(CS(=O)(=O)CCO)NC1(CC=C)CN(C(=O)CNC(=O)OC)C1 CCCCC(O)CC(=O)N(CCCNC(=O)C(N=[N+]=[N-])C(C)C)C CCC(CCC(=O)N(CCOC)C(C)C1CC1)NC(=O)C(F)n1ccnc1 C(C(C)C(=O)NC(C)(C)C(C)NC(=O)CCN(C)CCO)OCC N1(c2ncc(C(=O)OC)nc2)CC2CCC(NC(=O)C(=O)NC(C)C)CC2C1 Cc1cnc2n1CCN(C(C1CN(C)CCN1C(=O)COCCF)=O)C2 N1(C(Cc2cc(C)on2)=O)CC(CNC(C2(CC(F)F)CC2)=O)C(C)(C)C1 C(=O)(C1=CCCCC1C)N1CCCC(NC(C(CC#C)O)=O)C1CC C1(S(C)(=O)=O)(C(N2CCN(C(C3CC(C#C)(O)C3)=O)C(CF)C2)=O)CCOCC1 c1(C(=O)NC2CC(C)N(c3ncc(C#N)cc3Cl)C2)cc2ccccn2n1 C(C(C)C(=O)N1CCCC1CC(=O)NCCCSCC)OCC C1(C(=O)NCC(C)(CO)NC(c2c(C)csc2)=O)CCN(C)S1(=O)=O N1(C(C2(C)CC2)=O)CCCOC(CNC(=O)CC2CSCCS2)C1 C#CCC(C)(C)C(=O)NC1CC=C(C(=O)N2CC(C)(C)C2COC)C1 C1(NC(CCOCCN(C)C)=O)CCS(=O)(=O)C12CN(c1ncnc(=N)[nH]1)C2 C(=O)(C1=NN2CCCN=C2N1)NCC1(CNC(=O)CSc2cccs2)CC1 C1(=CC(=O)NCC2C(NC(C(C)=C3CC3)=O)C2)CCC(C)CC1 C#CCC(C(=O)NCCc1n[nH]cc1C(=O)NOC1CCC1)C1CC1 C1(C(=O)NC(C)(C)CNC(=O)C(C2CCCCC2)N(C)C)Cc2cccc(F)c2O1 N1(C(COCC(=C)C)=O)CCC(CO)(CNC(c2ccc(F)cc2F)=O)CC1 c1(C(=O)OCC)nc(CNC(=O)NC2CCCC(C)O2)c2n1CCCC2 CCCCC(O)CCC(=O)N1CCC1CNC(c1ccccc1C1(C)CCO1)=O c1(C(=O)Nc2ncccc2Cl)cn2c(n1)CN(C(=O)Cn1ccnn1)CC2 C(C(=O)NCCN(CCc1ccccc1)C(C1CC=CCO1)=O)(C(C)C)OC c1(C(C(=O)NCC(CNC(C2CC3CCC2O3)=O)OC)=O)ccc(F)cc1F C(=O)(CC(C)CC(C)C)N1C(C(=O)OC)CC(n2cc(-c3cccc(F)c3)nn2)C1 N1(C(c2n(C)ccn2)=O)CC(CNC(c2cc(CO)on2)=O)CC12CCOCC2 n1(CC)ncc(C(=O)N(C)CC2(NC(C3(C(C)C)CCCO3)=O)CC2)c1C1CC1 C1(C)(NC(C(C2CCOCC2)OCC)=O)CCN(C(=O)C=Cc2cncs2)C1 c1(OC)cc(C(=O)NCC23CC(NC(C4CC4CCN(C)C)=O)(C2)C3)ccc1OC C(=O)(CC1=CCN(C)CC1)N1CCC(CN(C(C=CC(CC)=CC)=O)C)C1 Cc1[nH]c(C#N)cc1CN1CC(NC2CCCC(C)CC2)C1.c12ccccc1O2 C(=O)(C#CC1CCCCO1)N1CCC(NC(C2C3CCCC23)=O)C(F)C1 CCC(N=c1ccc(Br)c(S(=O)(=O)NCC2CCCC2(C)C)[nH]1)c1cccnc1 c1(C(C)C)cnc(O)c(C(N2CCC2CNC(=O)Cc2cncnc2O)=O)c1 CC(CN(C)C)CCC(=O)NC(CNC(c1cc(C(F)(F)F)ccc1F)=O)CO c1(CN2CCN(C(CSC)=O)C(CO)C2)ccc([N+](=O)[O-])cc1Br C#CCCC(O)C(=O)N1CCCC(CNC(=O)CCn2nc(C)nc2C)CC1 C1(CN(C(c2ccc(C(N)=O)o2)=O)CC)CCCCN1C(C1COC(=O)C1)=O C(=O)(CCCC(F)(F)CO)NCC(C(C)C)NC(Cc1n[nH]c(=NCC)s1)=O N1(C(C2C(C)(CC)C2)=O)CCC(O)(C2(NC(=O)CC(=O)N(C)C)CC2)CC1 c1(C(C(=O)NCC(CC(C)C)NC(=O)CC2(O)CC2)C)noc2ccccc12 N1(C(C(CC=C)(C)C)=O)CC(C)CN(C(=O)Cc2ccc(OCC)cc2)C(C)C1 n1(CCC)cccc1C(=O)NC1CCCC1CNC(C1CC(=O)CO1)=O c1(CSCCC(N2CC3C(CNC(C(C)N(C)C)=O)C3C2)=O)ccc(C#N)cc1 c1(C(N2CC(NC(CC3(C(=O)OC)CC3)=O)C2)=O)cc(C(F)F)[nH]n1 N1(C(CC2C(C)C2)=O)CCN(C(c2cc(Cl)c(N)c(Cl)c2)=O)CC2(CC2)C1 n1(CCC)cc(Br)ccc1=O.Cc1cccc(-c2cn(CS(CCN)(=O)=O)nn2)n1 C(=O)(CCCCCN(C)C(C1(OC)CC1)=O)NCc1c(CC)nn[nH]1 C1(NC(Cc2ncn(C)n2)=O)CC(CC(=O)NCC2(C3CCC3)CC2)C1(C)C C(=O)(CC1=CCCC1)NCCCCC1(NC(c2cc(C)no2)=O)CC1 N1(C(N(C)Cc2csc(C(F)(F)F)n2)=O)CCOC(C)(C)C1C1CC1 CCCCC(CNC(=O)CCc1cccc(C(F)F)c1)NC(c1nncs1)=O c1(C(N2CCC3CC23C(=O)NCCF)=O)cc(F)cc(F)c1 c1(OC)cc(C(=O)Nc2ccc(CN3CCOC3=O)cc2)cc(C#N)c1O N1(C(C(CCC)NC(N)=O)=O)CC2CC(NC(c3cc(C)nc(O)n3)=O)C1C2 C1(CCNC(CC2CC(=C)C2)=O)CCCN(C(=O)C=CSC2CCOCC2)C1 N1(C(c2cnn(CC(F)F)n2)=O)CCC2(CCCN2C(C2CC3C=CC2C3)=O)C1 N1(C(c2c(OC)c(O)nc(O)n2)=O)CC(C)OC2(CCN(C(=O)CC#N)C2)C1 Cc1nn(C)c(Cl)c1CC(=O)NCC1C(C)CCN1C(=O)C=Cc1cccs1 CN1CCC(C(=O)N(CCCCN(C(=O)CSc2nnnn2C2CC2)C)C)C1 N1(CC)N=C(C(=O)NC2(COC)CCN(C(=O)C=C(C)C(C)(C)C)C2)CCC1=O c1(CC)cc(F)ccc1C(=O)NCCCCCN(C(=O)CSc1nnnn1C)C CC(CNC(C1(CO)CCCN(C(=O)C(O)C(F)(F)F)C1)=O)CC(F)(F)F Cc1cccc(CC(=O)NCC2CC(CNC(C3CC(O)C3)=O)CO2)c1Br C1(CNC(C=CCCC)=O)CN(C(c2ccc(C)c(Br)c2)=O)C(C)(C)C1 C1(NC(c2cccn3nncc23)=O)CCN(C(=O)Cc2cnsc2)C12CCCC2 S(=O)(=O)(c1cc2nc(O)[nH]c2cc1Br)NC1(C)CCCOC1 C(CCCCCCCC1CC1)(C(=O)NCCC#N)N(C)CC1C(C)C1 C1(C#N)(C(=O)NC(CCN(C(CSCCC)=O)C)C(C)C)CC2CC2C1 c1(OC)cc(OC)c(S(=O)(=O)NCC(=O)O)c(OC)c1.c12ccc(F)cc1SC2 C(=O)(C(CCF)NC(c1ncc(F)cn1)=O)NCC1(F)CN(C)C1 C(=O)(CC1CCCc2ccccc21)OC(C)(C)C.C12(C)CCCN1C(=O)C2C N1(C(c2cccc(SCC)c2)=O)CCN(C(c2ccc(N)c(N)c2)=O)CCC1C c1(C(N2CCC(C(C(=O)NC3CC(C(=O)OC)C3)C)C2)=O)[nH]cc(C)c1C C1(C(=O)NCCN(C(=O)CC2CCCC2)C2CC2)C2CCC1(c1ncco1)C2 N1(C(C(C)NC(N)=O)=O)CC2CCN(C(C3CCS(=O)(=O)N3C)=O)CC2C1 C(=O)(C#CC1CCC1)NCC(C1CCN(C(C(c2cccnc2)C)=O)CC1)(C)C C(C(CC(C)C)NC(c1cc[nH]c1C1CCC1)=O)NC(C(C)=CC1CC1)=O c1(OCC)ccc(C)nc1C(=O)NCC(C)(CC)NC(c1coc(C(N)=O)c1)=O Cc1c(C(N2CCCC(CC(=O)NOCCC(F)(F)F)C2)=O)ncn1C N1(C(c2c(Cl)cnc(CC)n2)=O)CCCC2CN(C(C3C4COCC34)=O)CCC12 Cc1ccc(CNC(C2C3CN(C(c4sc(OC(C)C)nc4C)=O)CC23)=O)cc1 C1(C2CN(C(C3CCN(C(C)=O)C3)=O)C2)(NC(c2cc(CC)ncn2)=O)CC1 Cc1cncc(CC(=O)N(C(C)CN(C)C(C2CC23CCCC3)=O)C)c1 Cc1cccc(F)c1CC(N1CCCC(NC(=O)C=Cc2cc[nH]n2)C1C)=O N1(C(c2cc(OC)c(F)cc2)=O)CC(NC(=O)CC(C)C(C)C)C2CCCCC12 CC(C)CC(C)CC(=O)NC(c1ccccc1)C(N1CC2(CC(CO)CO2)C1)=O N1(C(c2n[nH]c3c2COCC3)=O)CCC2CCN(C(c3snc(O)c3Cl)=O)C2C1 N1(C(C(C)NC(c2c(C)onc2)=O)=O)CCCC12CCCN(C(=O)CN(C)C)C2 C1(NC(COC(CNC(CCSCC)=O)(C)C)=O)CC2(CCC2)C1O.C(C)C C1(C(=O)NC2(CSC)CCC2)CC(NC(=O)C(=O)NC(C)C)CCO1 c1(C(=O)NC(CCNC(c2c(O)ccc(OC)c2)=O)(C)C)cc(F)c(F)cc1F C1(NC(C=CC)=O)CN(C(=O)COc2cccc(F)n2)C2(CCOC2)C1 c1(OC2CC(NC(c3ccn(C)n3)=O)C2)cccc(NC(=O)NCC(F)(F)F)c1 N1(C(c2n(C)cc(N)c2)=O)CCC2(COC(=O)N2)C1 c1(C(c2n(CCC3(C)CC3)nnn2)NC2(C)CCSC2)cc(Br)c(F)cc1F C1(NC(C(CN(C(=O)CCCn2cccc2)C)(C)C)=O)CCN2CCCCC12 C#CCC(C(=O)N1CCOC(CC)C1)NC(=O)CN1CC=CC1 C1(C(=O)NCCC(=O)OCC)(CNC(c2ccn(CC)c2C)=O)CCCCC1 N1(C(c2c(CC)nns2)=O)CCCC1C1CCCCN1C(c1csc(C)n1)=O CCCCCCCCC(=O)NCC1CCN(C(=O)Cc2ncccc2C)C1 N1(C(c2csc(Br)c2)C(=O)NCCCCCC)CCCCC12CCN(C)C2 O=S(=O)(c1c[nH]ccc1=NCc1n[nH]c2c1CCCC2)NCC1CCCCC1O N1(C(COCc2c(C)ncs2)=O)CCCC(C)(C)C1CNC(=O)C(C)(C)O c1(SC(C)C(=O)NC(C)C(CO)N(C)C)ccccc1.C12(CCCO1)C(=O)NC2 c1(C(=O)NC2COCC2NC(c2ccc(CO)o2)=O)cnc2c(c1)CCOC2 N1(C(C2C(OC)CCC2)=O)CCCC(NC(C2CCC(=O)N2)=O)CCC1 C1(CN(C(COC)=O)C)CCN(C(c2n[nH]cc2C2CC2)=O)C1 N1(C(c2c(C)sc(Br)n2)=O)CCC(C)C(CNC(c2coc(O)n2)=O)C1 Cn1nc(C(N2CCOC(C)(CNC(c3csc(O)n3)=O)C2)=O)ccc1=O CCS(=O)(=O)Cc1cn(CC2CCCN2C(C2(C)CC2C)=O)nn1 C(CN=c1[nH]c(=NC2CCCC(CC)CC2)[nH]c2c1SCC2)SCC=C C12(C(=O)NC3C=CCN(C(C(C)OC4CCCC4)=O)C3)CCN(CC1)CC2 N1(C(C)C)C(=O)CC(C(=O)NCC(=O)COCC(F)(F)F)C1c1ccc(Cl)c(F)c1 N1(C(c2cnc(OC)nc2)=O)CCCC(C)C1CNC(c1ccc(C)c(O)c1)=O c1(C(=O)NCC2(C)CC2c2ccccc2)cc(C(F)F)ccc1Cl CC(CCS(C)=O)NC(c1ccnn1C1CNC1)=O N1(C(CC(C(F)F)NC(c2cc(OC)ncc2)=O)=O)CCOc2ccccc21 c1(C(=O)NC2(C)CCN(C(=O)CCC3CCC3)C2)ccc2nc[nH]c2n1 C1(N(C(C2ON=C(CC)C2)=O)C)Cc2ccccc2C1 C(=O)(C1=Cc2ccccc2C1O)N(C)CCN(C)C(c1ccnc2ncnn12)=O c1(C(=O)NC2C=CC(CNC(CCCCC)=O)C2)cc(Br)cnc1N C(=O)(C(C)(C)C(C)O)NCC(CC)NC(=O)Cn1cccnc1=O N1(C(c2nc[nH]c3nccc2-3)=O)CC2CCN(C(C3CCCC3O)=O)CCC2C1 c1(CC(=O)N(C)CC2OCCN(C(CCCSC)=O)C2)ccccc1S(C)(=O)=O Cc1cnc2n1CCC(C(=O)NC1CCC1CNC(=O)CCN1CCCCC1)C2 C1(C(=O)N(O)CC2CCC(F)(F)C2)(c2ccccn2)CC2(CC2)C1 CCC(C(=O)NC(CNC(C1(C(F)(F)F)CC1)=O)CCOC)C(F)(F)F c1(C(=O)NC2CN(C(CCCn3ncc(C)c3)=O)CC2C)ncnc2c1CCC2 C1(NC(C2C(C(N)=O)C2)=O)CC2CC1N(C(c1cncc(C(F)F)c1)=O)C2 N1(C(C(F)=CC)=O)CCC2(CC1)C(OC)CC2NC(c1ccc(C2CC2)cc1)=O C(CC)(CCC(=O)NCC(C)(C)CCO)NC(C(CCC)F)=O c1(OCC(=O)NCC2(NC(C(CC#C)C)=O)CCCC2)cccc(C#C)c1 S(=O)(=O)(c1ccc(C(N)=O)cc1)NC(C(c1ccc(C)s1)C)=O CC(C(=O)NC1(CCCNC(=O)C(C)O)CC1)OCC1CC1 C1(C(=O)NC(C(C)C)(C)CNC(=O)Cn2cccn2)CC2CCC1NC2=O c1(C(=O)OC)ccc2c(CN3CCN(C(C4CN(C)C4)=O)C4CC34)c[nH]c2c1 C1(NC(CCc2cncc(C)c2)=O)CCN(C(=O)COCC2CCC2)CC1O Cc1c(N)ccc(C(=O)NC2(CO)CCN(C(=O)C(C)N3CCC3)CC2)c1C CCC(CC)(C(=O)NCC(C1CCC1)NC(=O)C=CSc1nc[nH]n1)OC c1(CCC)[nH]ccc1C(=O)NC1CC(F)(CNC(c2coc(CO)c2)=O)C1 C(=O)(C(C)(C)CNC(C1CCC(F)C1)=O)N(CC#CC)CC#C c1(C(=O)NCC(C2CCCO2)OC)sc2c(c1Br)CNC2 C12(NC(CSc3nc(C)[nH]n3)=O)CCCC(CN(C(C3(C)C=CCC3)=O)C1)C2 N1(C(C2(CCNC(C(C)SCCCC)=O)CC2)=O)CC2(CCC2O)C1 N1(C(C=Cc2ccc(SC)s2)=O)CCC(C)C(CNC(c2cc(SC)no2)=O)C1 c1(C(N2CCCCC2Cn2cc(C3CC3)nn2)=O)ccc2cc(O)ccc2c1 c1(NCCNC(CNC(c2cc(F)ccc2F)=O)=O)ccc(F)c(Cl)c1F c1(OC)ccc(C(=O)N(CCC(C)NC(C2(C)CCCCO2)=O)C)c2[nH]ncc12 c1(C(N2C(C)CN(C(C3CCC(=O)O3)=O)CCC2)=O)cc2n(n1)CCNC2=O c1(CCC)cc(C(=O)N(C2CCN(C(C3CCCCO3)=O)C2)CCC)nn1C c1(C)ccc(C)cc1F.N1(OCC)CCC(C)(CCO)C1 C1(C(=O)NCC(C)CNC(C2CC3(C2)CC(O)C3)=O)COCC2(CCC2)O1 c1(C(N2CC3C(CNC(c4ccsn4)=O)(C3)C2)=O)cc2c(nc1O)CCCC2O c1(OC)ncc(C(=O)N(CCC(C)NC(=O)C(COC)N(C)C)C)cn1 c1(C(N2CCC3(NC(CCCCOC)=O)C(C2)C3)=O)cc2cc(F)cc(F)c2[nH]1 c1(C(N(C)CC2CCCCN2C(c2csc(C(N)=O)n2)=O)=O)occ2c1CCC2 N1(C(CC2N(CC)C(=O)CC2)=O)CCOCC(CNC(=O)CC(C)(C)C2CC2)C1 C(N=c1[nH]cncc1I)C1N(C(CNC2(C)CCN(C(C)=O)C2)=O)CCCC1 c1(OC)cc(N)c(F)cc1C(=O)CN(C1(C(=O)NC(C)(C)C)CC1)C(=O)C1CC1 c1(C(=O)NCC(CN(C(C(CC)N(CC)CC)=O)C)O)ccc2c(cnn2C)c1 C1(C(N(CC2N(C(CC(C(=O)OC)C)=O)CCC2)CC)=O)CCn2nncc2C1 c1(CC)ccc(OC)c(-c2ccc(NC(c3nccnc3C(N)=O)=O)c(F)c2)c1 CCC(N=c1[nH]c(=NCC2(S(C)(=O)=O)CC2)[nH]c2cc(C)ccc12)c1cccs1 N1(C(C(C=C)c2ccccc2)=O)CCN(CC(=O)NCc2cc(C)c(Cl)s2)CC1 CC1CC2(CC(C(N3CCCC(N(CCF)C(c4ccc(=O)oc4)=O)C3)=O)C2)C1 O=C1NCCCc2occ(C(N3CCC3CNC(c3cncc(Cl)c3)=O)=O)c21 N1(C(C(CC)C2CCOCC2)=O)CC(NC(=O)C(C)Cc2cnc[nH]2)C(C)(C)C1 C1(NC(COCC#C)=O)CCN(C(=O)CN2CCC(C)CC2)CCC1CO N1(C(Cc2ccc(C)o2)=O)CCC(O)C(NC(=O)C(O)CC(N)=O)C1 CC1(C)CC2(CC(C(=O)NC3CN(C(c4cccc(F)c4O)=O)C4CC34)C2)C1 Cc1nn(C)c(Cl)c1C=CC(N1CC(NC(c2sc(Cl)cc2Cl)=O)C(C)C1)=O C(CCCC(=O)NC(C)CC(C)NC(c1ccccc1C(F)F)=O)OCC C1(C(=O)NC(C2CN(C(=O)C(C)(C)C)C2)C)CC2CC1C1C2C1(F)F c1(C(=O)NC(C2CCCCN2C(c2cscc2C(F)F)=O)C)n[nH]c2c1CCC2 N1(C(c2cccc(N(C)C)c2)=O)CC2CC(C1)CN(Cc1cc(Br)ncc1Br)C2 C1(CNC(CC(C)(C)OC)=O)CCC2(CN(C(c3sc4cncn4c3C)=O)C2)O1 C1(C(=O)NCCN(CCOC)C(C2CCC2c2ccc(F)cc2)=O)CCC(=O)NC1 c1(NC(=O)Cc2ccc(OCC(F)F)cc2)ncnc2c1COCC2 c1(C(N2CC=CC(NC(c3ccnc(OC)n3)=O)C2)=O)ncc2cc(Cl)ccn12 Cc1ccc(C(=O)NC2CCCCC2CNC(C2CC2(F)F)=O)cc1 N1(C(C=C(C)C)=O)CC2CCCC(CNC(C3C4CCCCCCC34)=O)C2C1 c1(C(=O)NC(CCOC)CNC(=O)CCC2CCCO2)cnc2cc(C)[nH]c2c1 N1(C(C(CC)OC)=O)CCC(C(=O)Oc2ccc(F)nc2)(OCC)C1 C1(C(=O)NC2CCN(C(CNC(=O)CC(F)(F)F)=O)C2)COCC2(CCC2)O1 C#Cc1cc(C(=O)Nc2cnn(CC(F)(F)F)c(=O)c2Br)cc(I)c1 C(=O)(CC(C)C(F)F)NCCCN(CCCNC(C(CC)OCCOC)=O)C CC(CC(=O)NCC1CC(NC(C2CC(F)CN2C)=O)C1)C(C)(C)C Cc1cc(C(=O)OC2CCCC(C(F)F)C2)ncn1 c1(CC(=O)NCC(CC(C)C)NC(c2cccc(=O)o2)=O)cccc([N+](=O)[O-])c1 C1(CC)C(C(=O)NCc2ncoc2C2CC2)CCN1C(=O)CCN(C)C(C)=O C1(C(=O)NC2C(NC(C(n3ccc(C)n3)(C)C)=O)CCOC2)CC12CC(C)(C)C2 c1(NC(c2ccc(SC)cc2)=O)ccc2nc(O)n(C3CC3)c2c1 C(=O)(CCCN=c1nc2c(cnn2C)c(NCCCC2CCCC2O)[nH]1)NCC c1(C(=O)NC2C(NC(c3scc(C)c3C)=O)C2)ccc2cn(C)nc2c1 c1(N(C)Cc2cc(OC)ns2)nc(C)cc(=NCC2CNC(=O)C2(F)F)[nH]1 CS(=O)(=O)c1ccnc(N2CCSCC2C(=O)NCc2ccccc2I)n1 Cc1cnc(Nc2cccc(CO)c2)nc1C(=O)N(CC(=O)N(C)C)C c1(NCCCSCC)ccc(S(=O)(=O)NC(c2ccoc2)C)cc1F c1(CC(=O)NCC(C)(CO)NC(c2cccnc2C(F)(F)F)=O)cncnc1O c1(C(N(C2CCCN(C(C3C=CCCC3)=O)CC2)CC)=O)cccc(F)c1OC Cc1nc(O)nc(S)c1C(=O)N(CC(O)CNC(C1CCn2ncnc2C1)=O)C C(CCN=c1[nH]c(=NC2CCC(C3CC3)C2)c2ncccc2[nH]1)OCCO c1(C(=O)NC2CC3CC2N(C(c2sccc2F)=O)C3)ccc2cnnc(O)c2c1 N1(C(C=CSC)=O)CCC(C2CCN(C(c3c(C)nsc3Br)=O)C2)C1 C(=O)(CC(C)(C)C(=O)NCCC1CCC(NC(c2c(C)nc(C)n2O)=O)C1)OC C(=O)(CCCC(=O)NC)NCC.C(C)(CCN)N(C(C1(CCCC)CC1)=O)C O=C(CCC(CF)CF)NCC1(CO)CCN(C(=O)C(C2CCOCC2)F)CC1 n1(CC(=O)NCCN(C)C(C2CCC3C2C3(F)F)=O)nnc2ccccc12 C(c1c(C)noc1C)=CC(=O)NCCOC1CCN(C(C2(CC)CC2)=O)CC1 C1(NC(c2cc(CCC)[nH]n2)=O)CC2(C1)CC2C(=O)N(C)CC1(C)CCC1 C1(NC(CCCN=[N+]=[N-])=O)CC1C1CCCN(C(C2(C3CCC3)CC2)=O)C1 Cc1ccc(C=CC(=O)NC2CCOCC2C(=O)NC2C3CCCOC23)cc1 C(C)(C)(CCC(=O)NCCC(F)=C(F)F)NC(C)=O CC(C(=O)NCC1CCCC1NC(C1(F)CC1)=O)C(=O)N1CCOCC1 CC(CC1CCCC1)C(=O)N(C)CCNC(c1cc(Br)sn1)=O C1(C(N(CCCNC(C2(F)CCOC2)=O)CC)=O)CCOC2(CCC2)C1 Cc1cn(C)nc1C(=O)NCC=CCC(=O)NC1C2CCCOC12 C(c1ccncc1)=C(C)C(=O)NC1CCC(NC(c2nonc2N)=O)CC1 c1(C(C)C)cccc(C(=O)N(C2CCN(C(C3(CF)CC3)=O)CC2)C)n1 N1(C(CN(C(C)C)C)=O)CCC2CCN(C(=O)Cc3csc(Br)c3)C2C1 S(=O)(=O)(c1cc(Br)cnc1Cl)NC1CC(C)(C)C(=O)NC1 O=C(C1=C(Cl)CCCC1)N1CCN(C(c2cnsc2)=O)C(c2ccncc2)C1 c1(C2(CNC(C(=O)N(C(C)C)Cc3ccco3)=O)CCCC2)cccc(Cl)c1F CC#CCCCC(=O)N1CCN(C(c2ccc(OC(F)(F)F)cc2)=O)C2CC12 S(=O)(=O)(c1ccc(C#N)cc1)N1CC2(C(=O)OCC)C(C1)CS(=O)(=O)C2 CC1=CCCN(C(N2CCCC2CC2CCCC2)=O)C1 C(=O)(C1=NNC(=O)CC1)NCC1C2N(C(CN(C(=O)OCC)C)=O)C(CC2)C1 C(C(O)C(=O)NCCCc1cn(C2CCOC2)nn1)=CC C(=O)(C(C)CC1CCC1)NC1CN(C2CCC2)C1.C12CC1C(=O)NC2C c1(CC(N2CCC2C)=O)ccc(F)cc1.C1(C(=O)OC)CCC(CN)C1 C(=O)(C(CCC(N)=O)n1cc(-c2ccc(F)c(F)c2)nn1)NC(COC)COC c1(OC)ccc(C)c(CNC2CCCC(C(N3CCC(C#N)CC3)=O)C2)c1 C1(NC(Cc2cnc(C)s2)=O)CCCN(C(=O)Cc2ccc(Cl)c(F)c2)C1C c1(C(N(CC(C)O)CCNC(C(C)OCC#C)=O)=O)cccc(OC)c1C N1(C(c2c(CNC(C(C)OC)=O)n[nH]c2)=O)CCCC(C)C1CO CC(O)C(C)(C)C(=O)NCC1CN(C)CCN1C(=O)CSc1nnnn1C N1(C(c2n[nH]c(CC)c2F)=O)CCC2(C1)CN(C(c1c(F)cc(Cl)cc1F)=O)C2 CC1CCCC(C)N1C(c1ccc(NC(=O)CCCNC(N)=O)nc1)=O N1(C(C(CCCC)O)=O)CC2(CCCCN(C(c3cnn(CC(C)C)c3)=O)C2)C1 C1(C)(CNC(C(C)OCC(F)(F)F)=O)CCN(C(=O)Cn2ncnn2)C1 N1(C(CC)=O)CCC(NC(=O)C(=O)Nc2cccc(CSC3CC3)c2)C(C)C1 N1(C(c2cn(CCC=C)nn2)=O)C2CCC1CN(C(c1ccc(C#N)s1)=O)CC2 C1(NC(c2c(OC)csc2)=O)CC2C(NC(=O)CCCF)C2C1 N1(C(Cc2scc(C)c2)=O)CCC2CCN(C(=O)C(C)(C)c3cscc3Cl)CC12 N1(C(CCC2(NC(CSCCCC)=O)CCC2)=O)CC2CC2(CC)C1 C1(C(=O)NCCCC#C)CC(N=[N+]=[N-])CN1C(=O)CC(C)C N1(C(CC(c2c(C)n[nH]c2C)C)=O)CCC2(C1)CN(C(=O)C(=O)N(C)C)C2 C(=O)(CCCC(C)=O)N(c1ccc(Nc2c(NC(C=C)=O)n[nH]c2)nc1)C C1(CC(=O)NC)CCCCN1c1ncccn1.C12CCCN(C1)N1CC(C1)N2C.CCO c1(C(=O)NC(C2(O)CCN(C(c3cc(C)c(C)[nH]3)=O)C2)C)cnc(O)c(F)c1 CC1(C)CN(C(=O)C2=CCN(C(C3(CO)CCCO3)=O)C2)C2CCCC12 N1(C(C2(COC)CC2)=O)CC(C)N(C(=O)CC2CCC(C)CO2)C(C)C1 Cc1cc(=N)[nH]cc1C(N1CCC(NC(=O)CC2CC3CCC2CC3)C1(C)C)=O C1(OC)CC(C(=O)NCC2(C3CC3)CC2)N(C(C)=O)C1 N1(C(C(C)NC=O)=O)CC2(CC(CC(=O)N(C3CC3)Cc3nncn3C)C2)C1 c1(NC(C2C(Nc3c(C)cncn3)C2)=O)cc(F)cc(I)c1 N1(C(c2cc(CCC)[nH]n2)=O)C2CC1CN(C(c1ccnc(CN(C)C)c1)=O)C2 CC1CCCC=C1C(=O)N1CCC(C(=O)NCc2noc(C3CC3)n2)O1 n1(C(C(=O)NCCCN(C(=O)CC2CCC3CC23)CCC)C)ccnc1CC N1(C(=O)C2CC2)CCN(C(=O)Cc2csc(Br)n2)C2CCCCC12 C1(C(=O)NC2CC(CNC(C3C4COCC34)=O)C2)CC2CC1C1C2C1(F)F c1(C(N2CCCC(N(C(CCSCC)=O)C)C2)=O)cc2c(O)cccc2[nH]1 c1(CNC(C(C)NC(C)=O)=O)ncoc1CCNC(=O)COc1ccccc1 C1(NC(C2(CCOC)CCC2)=O)CC(O)CN(C(c2coc(Br)n2)=O)C1 c1(CN2CCCC(CN3CCCC(C(=O)OC)C3)C2)ccc(C#CCO)s1 N(C)(C(=NCCC1CCCS1)NCCF)Cc1ccc(CC)cc1 Cc1cccc(C(=O)NC(CC2CC2)C(=O)N(C2CCNC2=O)C)c1O Cn1ccc(C(N2CC=CCC2C(N2CCCC(C)(CO)C2)=O)=O)cc1=O c1(NC2CN(C(c3cncc(Cl)n3)=O)C2)ccc([N+](=O)[O-])cc1Br C1(C(C)C)C(=O)N1.C1(N(CC(C)C)C(C2CCCC2)=O)CCCCC1 C(=O)(CCS(C)(=O)=O)N1CCC(O)(CN(C(C(C)C(F)F)=O)C)C1 Cc1c(C(=O)NCCC(C)(C)NC(C2CC2C(F)(F)F)=O)ccn1C(C)C C1(CC=C)CC(O)CC(CNC(=O)C(c2ccco2)NC(C)=O)O1 N1(C(C2(CC)CN(C(C3COCCN3C)=O)C2)=O)CC2C(OC)C2C1 C1(C(N2C(C)CN(C(=O)COC3CCCC3)CC2)=O)CC(=O)c2ccccc2C1 c1(CCC(N2CCC(N(C(=O)CC3CCOC3)CC)C2)=O)cc(C)sc1C N1(C(c2ccccc2F)C)CC2(CCC(CNC(=O)C(C)(C)S(C)(=O)=O)O2)C1 Cc1cccc(-c2cn(-c3ccc(Cc4ccc(SC)cc4)cc3)nn2)c1C#N N1(C(c2n(CC)c(O)nc2)=O)CCC(C)C(N(C)C(c2cc(OC)nn2C)=O)C1 CN1CCN(C(C23CCC2C3)=O)C(CNC(c2cnnn2C)=O)C1 c1(C(=O)NC2CC(NC(C3(OC)CCCC3)=O)C2)cc(S(C)(=O)=O)oc1C C1(C(N2CC(C)C(O)C2)=O)CCNC12CCOCC2 C12(CNC(c3occc3C3CC3)=O)CC1CN(C(=O)Cc1ccnc(O)c1)C2 N1(C(CN(CCOC)C)=O)CCOC2(CCCN(C(C3CCC(=O)NC3)=O)C2)C1 n1(C(C)C)ccc(=NC(=O)C2C3CC(O)C(C3)N2C(c2cc(O)cc(=O)o2)=O)[nH]1 CC(C(C)(C)CO)NC(=O)C(C)(C)C1CCN(C(C2CCCC2F)=O)C1 c1(C(=O)OC)ccc(C(=O)NC2CCCC(NC(=O)CC3CC34CC4)C2)nc1 Cc1ccc(-c2ccccn2)cc1NCC1CC1NC(=O)OCc1ccccc1 CN1CCC(C)(C(N2CCOC(CNC(c3cnn(CCF)c3)=O)C2)=O)C1=O c1(C(N2CC3(CN(C(c4c(C)cco4)=O)C3)C2)=O)ccc2cccnc2c1 C1(NC(C(C)Cn2cccc2)=O)CCC(N(C(=O)COC2CCOC2)C)CC1 c1(CC=O)cc(Cl)c(Br)c(Cl)c1.CN1CCN(c2nnc(-c3ccccc3)n2C)C(C2CCCCC2)C1 N1(c2nccc(OC)n2)CCCC(C)(C)C1CNC(=O)CC1CC2CCC1CC2 c1(C(=O)NCCN(C(=O)CP(C)(C)=O)CCOC)nc2n(c1Cl)CCCC2 C(C)(CNC(=O)Cn1ccc(C)c1)(C(C)C)NC(c1ccc(COC)o1)=O c1(C(N2C(C)(COC)CC(NC(=O)C=CC3CC3)C2)=O)ccc2cncn2c1 C(=O)(C1CCCc2cc(O)ccc21)NC(C)CCNC(=O)CSc1nncs1 c1(OCC(C)C)ncccc1C(=O)NCCN(C(c1cnnc(O)c1)=O)C(C)C c1(C(N(CC(C)NC(CCC2C(C)=NOC2=O)=O)C)=O)c(C)nn2ccccc12 CCCC(C)(C)C(=O)NCC(C)(C)CNC(c1cc(-c2cccs2)on1)=O c1(C(N(C(C)(C)CO)Cc2cccc(OCC)c2)=O)cnc2sc(Br)cn12 c1(C(=O)NCCN(C(c2c(Cl)ccc(NC)c2)=O)C)cc2ccccc2nc1OC C1(C(N2CCC(F)C(F)C2)=O)(CC)CCCN(C(=O)CCCC2CC2)C1 N1(C(CCOC)=O)CC2C(CNC(c3c[nH]nc3C(C)(F)F)=O)C2C1 c1(C(N2CC(CNC(=O)CCc3cncs3)C(F)(F)C2)=O)ccc2nncn2c1 CCC1=NOC(CN(C(=O)NC(C)(Cc2ccccc2)C(F)F)C2CC2)C1 c1(C(N(C(C)C)CCNC(c2cc(C(F)F)n(C)n2)=O)=O)cnc2n1CCC2 Cc1c(C(=O)NCCCOCCCNC(=O)C(C)C(C)C)sc2ccc(F)cc12 c1(NC(CC(CC)N(C(=O)CC2CC=CCN2C)C)=O)ccc2ccccc2c1 c1(C(N2CC(C)C(CCNC(=O)OC(C)(C)C)C2)=O)ccnc2[nH]c(O)nc12 CC(C)(CCC(=O)NCC(C)(C)NC(C1CCC(C2CC2)C1)=O)N1CCOCC1 c1(C(=O)NC(C2CN(C(=O)COC3(C)CCC3)CCO2)C)ccc2nnnn2c1 N1(C(CC(CC)C(C)(C)C)=O)CCN2CCN(C(=O)C(C)CC(N)=O)CC2C1 C1(C)(C(=O)NCCC2CN(C(C3C(c4n(C)ccn4)OCC3)=O)C2)C=CCCC1 n1(CC(=O)NC(C(=O)OC)CO)cc(Br)c(=O)c(I)c1 C1(C(=O)NCc2c(CC)nns2)C(C2CC2)CCN1C(c1ncn(CC)n1)=O CC1CN(C(=O)CCc2ncco2)CC1NC(C1(n2cccn2)CCC1)=O C1(CN(C(c2coc(C(C)=O)c2)=O)CC)CCN(C(c2ccn(CC)n2)=O)CC1 C#Cc1cnn(CC(=O)NC2C3CC(NC(c4cncc(N(C)C)c4)=O)CC23)c1 C1(OCC)CC(NC(=O)CC(C)c2ccncc2)C1OC C1(C(C)NC(=O)CSc2nc[nH]n2)CCN(C(C2(CO)CCCCC2)=O)CC1 C1(C(=O)NC2(COC)CC2)CC12CCN(C(=O)Cc1sccc1C)CC2 Cc1ccc2c(c1)CC(C(=O)NCC1CC(NC(=O)Cc3ccc(F)cn3)C1)S2 C(CCC(O)C(=O)NC1CCCCC1CO)NC(c1cn(C(C)C)nn1)=O N1(C(C(C2CN(C(CCC(N)=O)=O)C2)O)=O)CC2CCCC(O)C2C1 C=C=CCCC(=O)NC1COCC1C(N1CCN(C2CC2)CC1)=O CCCCCCC(=O)NCC1CN(CC(O)Cc2ccc(F)cc2)CCC1C c1(CC(=O)NCCC2(C(=O)OC(C)(C)C)CCC2)cccc2c1OCO2 c1(C(=O)OCC)cc(Br)c(C)cc1NC(N1CCC(O)(CN(C)C)CC1)=O C1(C)(OC)CCC(NC(=O)CC2(C)CCN2C(c2c(C)cncc2C)=O)CC1 C1(NC(CCCC#C)=O)CCC(C)N(C(=O)Cc2cncs2)C1 C(=O)(CC(CNC(C1(Cl)CC1(F)F)=O)OC)NC(COC(C)=O)CO c1(CCC(N2C(C(=O)NC3CONC3=O)CC(C)C2)=O)ccc2c(c1)OCO2 C1(NC(c2cc(C)nnc2)=O)CCC2(CCN(C(c3ocnc3C(F)F)=O)C2)C1 C(=O)(CC(C)(C)C(=O)OC)NC(C(=O)NCCOCCC)Cc1ccoc1 N1(C(CC(C)(C)C#N)=O)CCC2(CCOCC2)C(CNC(c2ccc[nH]2)=O)C1 N1(CC)CCC(OC(=O)NOCc2c[nH]nc2C)C1=O C(C(=O)NCC12CC1CN(C(C1(c3cccc(Cl)c3)CC1)=O)C2)(C(C)C)SC CC1CN(C(=O)C=CSc2nc[nH]n2)CCN(C(C2(CF)CC(=O)C2)=O)C1 C1(NC(CCCc2nc(C)sc2)=O)CC(C)CN(C(C2(C(C)C)CC2)=O)C1 c1(C(=O)NCC(CNC(=O)CCSC)OC)ns[nH]c1=O N1(C(CCCC=C)=O)CCC(C2(NC(c3cccc(=O)n3C)=O)CC2)C1 C(=O)(C1COc2ccccc21)N1CC(c2c(CNC(C(C(C)C)O)=O)nco2)C1 C1(NC(C2CCS(=O)(=O)N2)=O)C2CC3CN(C(C4C5CS(=O)(=O)CC45)=O)C1C3C2 C12(C(N3CC=CC(NC(c4cnc(Cl)s4)=O)C3)=O)CCCC1C2(F)F C1(C(N(CCOC)C)=O)CC(C)(C)CN1C(c1cccc(=O)n1C)=O C(CCCCCNC(C12CC1CCN2C(c1cn[nH]c1)=O)=O)N(C)C c1(CC(=O)N(CC(C)NC(=O)CN(C)C)CC)c[nH]c2ccc([N+](=O)[O-])cc12 c1(N2CC(C(C)NC(C(C(C)C)OC)=O)OCC2)nc(Cl)nc(C)c1F N1(C(CCCOC(C)(C)C)=O)CC=CC(NC(C2(CS(C)(=O)=O)CCC2)=O)C1 CC1CC(C(=O)NCCC2CCCN(C(=O)CC3=CCCCC3)C2)CC(C)(C)C1 C1(NC(COCC)=O)C(C)(C)CN(C(C2(CF)CC3(CCC3)C2)=O)CC1(C)C N1(C(C2CC(C)OCC2)=O)CC(NC(=O)Cc2ccco2)Cc2ccccc21 C1(NC(c2csc(Cl)n2)=O)CC2CC1N(C(=O)CC1CCOC1=O)C2 c1(CC)onc(C)c1C(=O)NCCC1(OC)CN(C(C2CN(C(C)=O)C2)=O)C1 C=CCCC(C(=O)NC1CCCN(C(=O)CCOCC(C)C)C1)c1ccccc1 C1(OC)CN(C(=O)CSc2nnc(S)s2)CC1NC(C1C=CCC1)=O C1(C(=O)NC2CC3CN(C(c4c(C)cc(F)s4)=O)CC32)CC2C(C1)C2(C)C N1(C(CN(C)C)=O)CC(O)(CCNC(C2CCN2S(C)(=O)=O)=O)C1 CC1(C)CCC2(CC1)CC2C(=O)NC1CN(C(=O)CNC=O)CC2CC12 c1(C(=O)NC(CN(C)C(c2cc(CO)[nH]n2)=O)(C)C)cccc(Br)c1N N1(C(C(C(=O)OCC)F)=O)CC(NC(c2sc(C)c(C)c2C)=O)CC12CCC2 CC(C)C(CCN(C(=O)C(O)Cc1cnc[nH]1)C)NC(C1CC1(C)C)=O N1(C(c2c(C)nsc2C)=O)CC(NC(=O)CC(C)O)C2(CC2)C1 N1(C(C2(N(C)C)CC2)=O)CCC2CN(C(c3ccnc(C4CC4)n3)=O)CC12 CC(C)(C)CCCC(=O)N1CC2CCN(C(=O)CCCCOC(C)(C)C)C2C1 c1(NC(C(c2nc(C)c(C)o2)N(CC(F)F)CC)=O)cccc(OC)c1 C1(OC)CCC(C(N2CC=CC(NC(=O)CC3CC3C(F)(F)F)C2)=O)CC1 C1(OCC(=O)NCC(c2ccccc2F)F)CCC(F)(F)CC1 CCC(C#N)C(=O)Nc1cccc(CCC(c2ccccc2)O)c1 C1(CC=C)(NC(c2cc[nH]n2)=O)CCN(C(=O)CSCC(F)(F)F)C1 c1(C(=O)OCC)c(F)cc(S(=O)(=O)OC2CCC(=O)N(C(C)C)C2=O)cc1F C1(CCC)CN(C(c2ccc(N)cn2)=O)CCN1C(=O)CC1CCCC(=O)N1 C1(COC)C2CC3C(C2N(CCCO)C(=O)Nc2cccc(OC)n2)C13 N1(C(C(C)NC(C(CO)OC)=O)=O)CCC(O)C1C c1(-c2ccc(NC3C4(CCC(OC)CC4)C3)s2)ccc2c(c1)OC(F)(F)O2 c1(C(=O)NC)cn(CC(N2CCC(C(O)C(F)(F)F)C2)=O)nn1 c1(C(=O)NC(CC)CCC(=O)NCC2(CCO)CCC2)n[nH]c2ccccc12 c1(C(N2C(CCNC(=O)CCCc3ccsc3)CCC2)=O)ccc(CCO)cc1 c1(C(=O)NC(CNC(C(CC)SC)=O)(C)CC)cc(C(C)(C)C)oc1C C(C(C)C)(C(O)C(=O)NCC1CCCCN(C(c2nc(=N)cc[nH]2)=O)C1)OC c1(CC(=O)Nc2c(Cl)ccc(OC)c2Cl)n[nH]c2cc(C3=CCCCC3)ccc12 C1(C(=O)NCC(C)(C)OC)CCN(C(=O)CCC2CCCN2C)CC1 c1(N(C2CC2)C(N(CCC(F)(F)Cl)C)=O)cccc(N2CC=CC2)c1 N1(C(C(C(C)C)=O)=O)CCN(C)CC1C(N1C(C)CCC1(C)C)=O CCCCCCCCC(C)C(=O)NC1CN(C(C23CCC(CC2)C3)=O)CCC1F c1(SC)ccc(Cl)c(C(N2CCCC(C)C2CCNC(=O)CCOC2CC2)=O)c1 N1(C(CSCCN(C)C)=O)CCCC(N(CCO)C(c2ccnn2CC#N)=O)C1 C(=O)(CCCCCF)NCc1c(C(=O)NC(c2cccnc2F)C)cco1 C(C)(C)(CCCC(=O)NC1CC(CF)C1)NC(CC1ON=C(CC)C1)=O C=CCC(C)C(=O)NCc1occc1C(=O)NCCCc1ccccn1 Cc1c(N)ccc(C(=O)NC2CCN(C(C3CCCC3(C)C)=O)C2)c1Cl C(CC(C(=O)NC1CC1(C)C(C)C)NC(C12CC(CO)(C1)C2)=O)=CC C1(NC(C(C(C)C)OC)=O)CCN(Cc2nc(C)no2)CC1O c1(OC)ccc(CC(=O)NC2CCC2CNC(=O)CC2CC3(COC3)C2)cc1 n1(CC(=O)NC2CC(F)(F)CC2NC(=O)CCC2CCC2)ccc2ccccc12 CCCCCCC(CC)C(=O)NCC1(F)CCCN(C(=O)CC2(C)CC2(F)F)C1 c1(C(=O)NC(C)CNC(C2CC2C(=O)OC(C)(C)C)=O)cc(Br)c2n[nH]cc2c1 c1(CC)cc(C(=O)NCC2CN(C)CCN2C(=O)Cc2nc(=N)[nH][nH]2)cc(F)c1 Cc1noc(-c2ccccc2)c1C(=O)NCC(C1CC1)N(C)C(C1CC1C)=O CC1=CCN(C(c2nc(C)c(C)s2)C(=O)NCCOC)CC1 c1(CC)nc[nH]c1C(=O)NCC1(CCNC(=O)COCCO)CC1.C1(C)CC1 O=C1CNc2cc(C(N3CC4CC(C3)N4)=O)cnc2N1 C(CO)(CCCCNC(C1(CF)CC(F)(F)C1)=O)NC(C1(C)CCCCO1)=O C1(NC(C(CC)=CC)=O)CCC2CCN(C(C3CCOCC3)=O)C1C2 C(CCC)(C(=O)NC(C)CC(C)NC(=O)C(C)NC(N)=O)=CCC c1(C(=O)NC(C2CC=CCC2)c2ccccc2)cnn2cnnc2c1 N1(C(=O)COCc2nc[nH]n2)CCOC2(C1)CN(C(=O)C(O)C1CC1)C2 CN1C2CCC1CC(=CC(N1CCC(NC(=O)C3CC3)C(C(C)C)C1)=O)C2 CCCC(CC)C(=O)N(CCCNC(=O)CC(C)c1ccccc1)C c1(NC(c2ncc(Cl)cn2)C)ccc(S(=O)(=O)NCC2(N(C)C)CC2)c(Cl)c1 c1(NCC(C2CCCCC2)NC(c2nn(C)c(O)c2)=O)ncnc2scnc12 c1(N(C(COC)COC)C)nc(N2CCSCC(C)C2)c2c(n1)CCCC2 c1(C(=O)OCc2c(Br)ccc(C(C)=O)c2)cn2cccnc2n1 N1(C(c2c(CC)nn(C)c2)=O)CC2(CCC(NC(C3CC(C)C3(C)C)=O)CC2)C1 c1(-c2c(C)nc(CC)s2)n[nH]c2ccc(C(=O)Nc3cccc([N+](=O)[O-])c3)cc12 c1(-c2c(C)occ2)nc(CCc2nncn2C)n(CCC(C)(C)C)n1 C1(C(=O)NCCC2(O)CN(C(c3ccc(CSC)o3)=O)C2)CCCN1C=O c1(C(N(C)CC2(O)CCN(C(c3cc(CC)no3)=O)C2)=O)ccc2cnoc2c1 CC(C)C(C)C(C)CC(=O)NCC1CCN1C(c1ccc2c(c1)ncn2C)=O c1(C(=O)NC2(C3N(C(C=CCOC)=O)CCC3)CC2)ccnc2c1cnn2C c1(C(N2CCCCC(CNC(C(C(C)(C)O)F)=O)C2)=O)cccc2sccc12 C(=O)(CCCC(C)(F)F)N(C)CC1(O)CCN(C(=O)CC2CCC(=O)NC2)CC1 n1(C(C)(C)C)nc2c(c1C(=O)NC1CCC1CNC(=O)CCCC#N)CCCC2 C1(C(=O)NCC2(NC(c3c(OC)nn(C)c3)=O)CCCCC2)CN2CCN1CC2 c1(C(=O)NCC(C)N(C)C(c2cc(O)ccc2Cl)=O)ccc([N+](=O)[O-])[nH]1 C12(C(=O)NCC(C(=O)NCCN(CC)CC)N(C)C)CCCC1C2(F)F C1(NC(c2cnc3c(c2)COC3)=O)CCN(C(=O)C(F)=CCCF)CCC1CO c1(CN2CCC3(CN(c4ccccc4)C3)C2)cnn2c1OCCCC2 C(CCCC(=O)NC1CCOC1C(N1CCC(CCCO)CC1)=O)OC C(=O)(C(F)(F)Cc1ccccc1)NCC(CO)NC(c1nc(C)oc1)=O C(CN=c1[nH]cc(C#N)cc1C)N(C(CNS(CCCC)(=O)=O)=O)CC C(=O)(C(C(=O)OC(C)(C)C)C(C)C)NC(CC)CNC(=O)CCc1cnc(C)o1 C1(SC)CCC(N=c2[nH]c(=NCc3c(Br)cnn3C)[nH]c3ccsc23)C1 N1(C(=O)CCCc2ncco2)CC2CC(C1)N2C(C12CCC(F)C1CC2)=O c1(OCC)ccc(CN2CCC2C(=O)NC(CCF)C(=O)OCC)cc1 C#CC1(C(=O)NC2CCC3(CC3)C2)CCN(C(C2Cc3nccn3C2)=O)C1 CCC(C)(C)C(O)C(=O)N(C1CCC(NC(=O)C(C)n2ccnc2)CC1)C c1(CNC(N2CC(C#C)OCC2)=O)nn(C)c(C)c1S(N)(=O)=O N1(C(c2c(C)onc2)=O)CCC2CCN(C(C3CC3CC(C)C)=O)C2C1 c1(OC)cc(F)cc(C(=O)NCC2(C(N)=O)CN(C(C3(C(F)F)CC3)=O)C2)c1N C(=O)(C(CCC)NC(C1CCC(=O)C1)=O)NCCC(=O)NCC#C C(=O)(CC(C)CC(F)(F)F)NC1C(C)N(C(c2cnc(=NCCF)[nH]c2)=O)CCC1 C(=O)(CC(C)CCC=C(C)C)NC1CN(C(c2nc(CC)oc2C)=O)CC12CC2 C(C(O)C(=O)N(C(c1ccccc1)CNC(=O)C=Cc1cn[nH]c1)C)=CC n1(CC(=O)NC(CC2CCCO2)C(=O)O)cc([N+](=O)[O-])cn1 N1(C(C(C)OCC)=O)CC(CNC(c2ncc(C(F)F)s2)=O)OC(C)(C)C1 Cc1noc(CCC(=O)NC2(CCNC(C3CC(F)(CO)C3)=O)CCC2)n1 CCC(O)C(C)C(=O)N1CCN(CCN(C)C(c2cc(Cl)cc(Cl)c2)=O)CC1 C1(C(=O)OCC)CCN(C(=O)CC2CCCN2C(c2cn(C)cn2)=O)C1C c1(SC)nc(C(=O)NC2(CO)CN(C(C3(CC(C)C)CC3)=O)C2)c2ccccn12 Cc1cc(C(=O)NC(CO)C(=O)NC2(CO)CC3(CCC3)C2)c(C)cn1 C(C)(N=c1nc2c(ncn2C(C)C)c(NCC2(C)CCC2)[nH]1)c1cc(C)on1 C1(CN(C(C2(CC#C)CC2)=O)C)CN(C(=O)C(CC)n2nccc2C)CC12CC2 CCC(C)C(=O)C(=O)NCc1cncc(C(=O)NCCSC(C)(C)C)c1 c1(CC)cnc2ccccc2c1C(=O)NCCC1CN(C(=O)COC(C)(C)C)C1 CC1Cc2c(C(=O)NCc3cccnc3Cl)cccc2CO1 C(=O)(C(O)CC(N)=O)N1CC(CCC)C(NC(C2CCCC23CCC3)=O)C1 Cc1cn(C)cc1C(=O)NC1(CNC(C2(C)CC2Br)=O)CCCC1 N1(C(c2c(CC)onc2C)=O)CC=C(C(=O)N(C2CCC2)C)CC1 c1(C(N2CCCN(C(C3C(=C)C3)=O)CC2)=O)cc2ccncc2o1 Cc1ccc(F)c(C(=O)NC2CC(S(C)(=N)=O)C2)c1Cl C=Cc1cncc(C(=O)NC(Cc2ccoc2)C(N2CCC(C)C(O)C2)=O)c1 Cc1ccc(-c2cc(NC(=O)CC(C)F)n(C)n2)cc1.N12CCC(C1)C2=O CCC(C)CCCC(=O)N1CC(O)CC1(C)C(=O)NCc1cnc(C)o1 C(=O)(CCP(C)(C)=O)N1C(C(N(CCC#C)CCOC)=O)CSCC1 N1(C(C2C(CC)C2)=O)CCN(C(c2ccc(C3CCCCC3)o2)=O)CC1C(F)F C1(NC(C(C)S)=O)CC2(C1)CC(NC(C1(c3ccccc3)CC1)=O)C2 CCC(C)C(C(=O)NC1(C(=O)NC(C)(C)CCCO)CCSC1)N(C)C CC1(C)CC(COC(c2sccc2C2CC2)=O)CO1 c1(COC)ccc(C(=O)NC(C2CCCN2C(=O)CC2CCC2)(C)C)cc1F N1(C(C2OCCO2)=O)CC2OCCN(C(c3ccsn3)=O)C2C1 N1(c2nnc(C)s2)CCC(NC(c2cccn3nnnc23)=O)C2(CCC2)C1 c1(C(N2CC(C)(OC)C2c2ccccc2)C(=O)NC)ccc(C2(OC)N=N2)cc1 C1(C(N2C(C)CN(C(c3nccn3C)=O)CC2)=O)CCOC2(CCCCC2)C1 C1(C(N(CCSC)CC)=O)C=CCN(C(C2CC(=O)CCO2)=O)C1 c1(C(=O)NCC2(CN(C)C(c3cnn(C(F)F)c3)=O)CC2)c2c(nn1C)CCC2 C1(CC=C)(C(=O)NC2CN(C(C)=O)C2)CN(C(C2CC2OC(C)(C)C)=O)C1 C1(CNC(c2cc(C)ncn2)=O)CCC2(CN(C(c3ccc(Cl)cc3O)=O)C2)O1 C1(c2n(C(C)C(F)(F)F)nc(-c3ccc(Cl)cn3)n2)CC12CC(F)(F)C2 CCC(C)(CNC(=O)CCCN=[N+]=[N-])C(=O)NCC(C)C(C)O C1(C(C(=O)NCC(C)CN(C)C(C2CCCCN2C)=O)F)CCCCCC1 c1(C(=O)NCC(N(C(C(C=CC)O)=O)C)C2CC2)cccc(C)c1Cl C1(COC)(NC(=O)COCC2CCCOC2)CN(C(=O)C=CC=C(Cl)Cl)C1 C1(F)(C(=O)NC2(C)CC=CCC2)CCN(C(C2(C)CC=CC2)=O)CC1 C1(F)(CNC(c2cnn(C)c2N)=O)CC(N=c2[nH]c(Cl)nc3[nH]ccc23)C1 C(=O)(C1Cc2c(Cl)cccc21)NC1(CCNC(CC2C(C)(C)CCCC2)=O)CC1 C1(F)(C(N2CCN(C(CN3CC(CC)C3)=O)CC2)=O)CCN(C)CC1 C(c1ccccc1F)=CC(=O)NCC1(NC(C2NC(=O)OCC2)=O)CCC1 C1(NC(C(C)SC)=O)CCCN(C(=O)C(F)(F)c2cncs2)CC1 C(CN=c1cc(CC2CCCCO2)nc[nH]1)C1N(CC(C2CC2)OC)CCCC1 C1(CNC(=O)NCC2CCCC(F)(F)C2)CC2(COCCO2)C1 Cc1cc(CN2CC(O)CC2(C)C)c(C)cc1O.C12CC1C(=O)N2 N12CCN(CC1C(F)F)C(=O)C1C(C1)C2=O.C1(C(=O)OCC)CC(SC)C1 C1(C(=O)NC2(CO)CCOC2)CC2(CCC2=O)C1.c12ccc(nc1)NC(=O)CNC2 c1(C(C(=O)N(C)CCN(C)C(c2ccncc2)=O)O)ccc(C#N)cc1 C1(CCOC)(NC(=O)CC2(O)CCCC2)CCN(C(c2ccc(CO)o2)=O)C1 CC1(C)CCCC(O)(C(=O)NC2CC(NC(=O)C(C)(C)C3CCCC3)C2)C1 Cc1nc2cc(CC(=O)NC3CCCCC3NC(C3CC3F)=O)ccc2o1 c1(OCCC(N2C3C(CNC(=O)C4CC4)C(C3)C2)=O)ccc(Cl)cc1[N+](=O)[O-] Cc1cccc(C)c1C(O)C(=O)N(CCNC(=O)Cc1nc(C)c(C)[nH]1)C1CC1 c1(CC(=O)NCC2(NC(C(c3c(C)cncc3)C)=O)CCC2)c[nH]c(=N)nc1O c1(C(=O)CCC(=O)Nc2ccc(-c3ncc[nH]3)cc2)ccc(Cl)cc1Cl N1(c2ccc(-c3c(F)ccc(C(=O)NC)c3)nc2)CCC(S(C)(=O)=O)CC1 CN1CCCN(C(=O)CCOCCCNC(c2cc(O)cc(=O)o2)=O)CCC1 C1(C(=O)NCC(c2cccc(Cl)c2)NC(=O)CCC(F)F)CC2(CCC2)CO1 C1(OC(C)C)CCCN(C(=O)C(C)NC(=O)Cc2ccsn2)C1 Cc1cc(C(=O)NCCCC(C)NC(C2(CF)CCC2)=O)cc(C)c1Cl C(=O)(CCC1CCc2ccccc21)NCC1N(C(c2cc(C)c(C)[nH]2)=O)CC=C1 C12(NC(CCOC)=O)CCCC1CN(C(=O)CC1CC3C=CC1CC3)C2 Cc1ccc(Br)c(CCC(=O)NCC(C)CNC(c2coc(C#N)c2)=O)c1 C(CCCC(=O)N1CC(CCNC(=O)CC2C=CCCC2)C(C)C1)OC c1(C(=O)NC(C(=O)NCC(=C)Br)C2(O)CCC2)nn(C)cc1Cl Cn1cnc2sc(C(=O)NCC(C)(C3CCC3)NC(=O)CSC(F)F)cc12 c1(C(N2CCC(N(C)C(=O)OC(C)(C)C)C2)=O)cccc(CN(C)C)c1 c1(NC(COC(CNC(c2c(OC)cnnc2)=O)(C)C)=O)n[nH]c2c1CCC2 C1(NC(CC(CC)C2CC2)=O)CN(C(=O)C(c2ccc(Cl)cc2)(C)C)CCC1F C1(NCC2CCC(OCCOC)CC2)CC2CCCC(Br)(C1)C2 C(C(C)C)(C(O)C(=O)N1CC(O)CC1C(=O)N(C(C)CC(C)C)C)OC CC(=O)C(C)CC(C)C(=O)NC(C(N1CC2CCC(CC2)C1)=O)C1CC1 C1(NC(C(Cc2ncn(C)c2)O)=O)CCN(C(C2(F)CCCCC2)=O)CC(O)C1 C1(NC(Cc2cncc(C)c2)=O)CCCCN(C(c2cn(C)c(O)n2)=O)C1 C1(C(N(C)Cc2ncc(C)o2)=O)CCC(CNC(C2COC(C)C2)=O)CC1 c1(C(COC(=O)C(C)(O)CO)=O)ccc(Cl)c(Cl)c1.CC1C(=O)N1 N1(Cc2nc(CCC)sc2)CCC(C(=O)NCc2cccc(CC)n2)CC1 C1(C)(C(N2C(C)CCC2)=O)CCN(C(c2cc(C3CC3)on2)=O)C1 N1(OC(c2cc(OC)c(F)cc2)=O)CC2(CC=CC2)C1C(C)C c1(CC(=O)NCCCCC(C)NC(C2(C)CCCS2)=O)ccc(Cl)c(F)c1 O=[N+]([O-])c1cc(C(F)(F)F)cc(Br)c1NC1CCCC2CC12 c1(C(=O)NC2CCN(C(C(C)OCCC#C)=O)C(C)C2)cccc2c1ncn2C C(c1cc2ccccc2o1)=CC(=O)NCC(CNC(C(C)(O)C1CCC1)=O)O Cc1ccc(C=CC(N2CCC(CCNC(=O)CN3CCC(C)(O)C3)C2)=O)o1 C1(C)(CNC(C2CCN(CCC)CC2)=O)CCN(C(C2CC(F)C2)=O)CC1 c1(C(C)(C)C)nc(C(=O)NC2CC(CCNC(C3CCCS3)=O)C2)co1 c1(CC(=O)N(CCCCCNC(C(COC)(C)C)=O)C)cccc2ccccc12 C12(C(N3CC(N(C(c4cc(C(=O)OC)no4)=O)C)C3)=O)CCCN1S(=O)(=O)CC2 N1(C(c2c(OC(C)C)cccn2)=O)CC2(CCCC2NC(C2CC2(F)F)=O)C1 N1(C(CC)=O)CCCC(NC(c2ccccc2-n2cc(Br)cn2)=O)CC1 C1(C(=O)NC2CCCC(NC(c3c(CC)scc3)=O)C2)CCc2nccn2C1 C1(NC(CCSCCCC)=O)CCC(Cn2cc(CC(=O)OCC)nn2)C1 N1(CC(=O)NC2(CC=C)CN(c3cc(Cl)nc(SC)n3)C2)C(=O)CN(C)C1=O C1(NC(C=C(C)Cl)=O)CC2CCCC(C1)N2C(=O)CC1(C(F)(F)F)CC1 C=CC1(C(=O)NC(CNC(=O)C(c2c(F)cccc2F)(C)C)CO)CCCCC1 C(=O)(CC1OCc2ncccc21)NCC1(C)CCN(C(c2cc(CO)[nH]n2)=O)C1 C12(C(=O)NCC3N(C(C4(C)N(C)CCC4)=O)CCC3)CCC(O)(CC1)CC2 c1(C(=O)NC(C2N(C(CCSCC)=O)CCCC2)C)ccc(C2CC2)nc1C n1(CC=C)nc(COC(C)(C)C)nc1CCN1CCCCC1 C(=O)(C1=CCCCCC1)N1CC2(C1)C(=O)N2.C1(CC)CCCCC1CC c1(C(=O)NC2CN(C(c3cccc(SCCC)c3)=O)C2)cn(C)c(=O)n1C c1(C(=O)NC2CC(NC(C3(Cc4ccccc4)CC3)=O)C2)cc(Cl)c(Cl)[nH]1 N1(C(CCC#N)=O)CC2(CC(NC(=O)C3=CC(O)CCC3)c3nccn32)C1 N1(C(C2C(C)(C)CC2)=O)CCCC2(CCN(C(C3(C)CC4CCC3C4)=O)CC2)C1 c1(CC)cc(C(N2CCN(C(C3CCCS3)=O)CC2CO)=O)ccc1OC c1(CC)ccc(F)cc1NC(=O)C(c1ccoc1)NC(=O)Cc1cn[nH]c1 C(=O)(C(CC(C)C)NC(=O)C1CC1)NCC#CCNC(c1cc(OC)ncc1)=O.O C1(C(N(C)CCNC(=O)Cc2nnc(C3CC3)o2)=O)CC2(C1)CC2(F)F Cc1nc2c(s1)CC(C(=O)NC1C3CCC1N(C(=O)CN1CCCC1=O)C3)CC2 CCCCCC(=O)N1CC(O)(C(C)NC(C2CCC(N(C)C)CC2)=O)C1 C(C(CC)C(C)(F)F)NC(C1N(C(c2n(C=C)ncc2)=O)CCOC1)=O N#Cc1ccc(C(=O)NCC2CC(F)CN2C(C2CCCS2)=O)s1 c1(C(N2CC=CCC23CCOC3)C(=O)NCCC2CC2)nc2c(s1)CCCCC2 C(C)(C(C)C(=O)NC)OCC1(C(=O)NC2(C(C)(C)OCC)CC2)CCC1 c1(C(=O)NC2CN(C(C3C(CCC)CCC3)=O)C2)cc2cc(C)cc(C)c2[nH]1 C(=O)(C1CSc2ccccc21)NC1COCCN(C(C2C(C(=O)OC)C2)=O)C1 C1(CNC(Cn2c(C)cc(=O)cc2)=O)CC2(CO1)CN(C(C1CC(C)(C)O1)=O)C2 CC1=C(C(=O)NC2CCC(C)(CNC(=O)Cc3c(F)cccc3F)C2)CCC1 C1(C)(C(=O)NCC(CC)NC(=O)CCCNC(=O)C(C)(C)C)CCCC1C C1(C(C)C)CN(C(=O)CC2CC(C)(C)CO2)CC1C(=O)NC(C1CCCC1O)C C#CC1(C(=O)NC(COCC)C(=O)N2CCC(CC)C2)CC(=O)C1 C(=O)(CCCCCCC(=O)NCC1CCN(C(c2coc(Cl)n2)=O)CC1)OC C1(C(N2C(Cn3cc(CN(C(C)=O)C)nn3)C=CC2)=O)CC2(CC2)CO1 C1(C(N2CC3C(C(=O)Nc4cc(CC)c(C)s4)C3C2)=O)CC(=O)N(OC)C1 C1(C(N2CCC(N(C(CN(CCC)C)=O)C)C2)=O)CC(C)N(C)C1 N1(C(C(CC)F)=O)CCC2(CCC(NC(=O)C(C)Cc3ccccc3)CC2)C1 C(=O)(C(CC)CCC)N(C)CC1CCN(C(COCCC=C)=O)CC1 c1(C(C(=O)C(COCCOCC)=O)(F)F)cccc(C(=O)NC2CC2COC)c1 C1(NC(=O)C=Cc2ccsc2)CC(CNC(=O)CNc2nccs2)C12CCC2 c1(C(=O)NC(CNC(C(C)SCC)=O)CCOC)cncc(Cl)c1 c1(CC(N2CCC(NC(c3c(C)cc[nH]3)=O)C(C)C2)=O)c[nH]c2cnc(Cl)cc12 N1(C(=O)CCCc2ccsc2)CCN(C(c2ccc(CO)nc2)=O)CC(CO)C1 C1(NC(C2(CNC(C(n3c(C)ncc3)C)=O)CCC2)=O)CCCCCC1F Nc1cc(CN2CCCCC2CC(O)C(F)(F)F)ccc1Cl c1(C(C)CNC(c2nnnn2CC2CCOCC2)C2CC=CC2)ncccc1F C(=O)(C(C)(C)C(N)=O)NC1CCCC(NC(C(C)c2ccco2)=O)C1 C1(CNC(C(C(=O)OC)(C)F)=O)CCN(C(=O)CC2CCOCC2)CC1C1CC1 c1(C(=O)NCC2CCC2(F)F)cccc2c1CNCC1(CC1)CC2 c1(C(=O)OCC)[nH]cc(C)c1C(=O)NCC1COCC1NC(C1(SC)CCC1)=O C1(OC)CC(C2CC2)N(C(=O)C(=O)NCc2ccc(N3CCCS3(=O)=O)cc2)C1 c1(CN2CC(C)(CNC(c3cc(F)c(Cl)c(F)c3)=O)C2)c[nH]c2cc(F)ccc12 Cc1cc(C(=O)NCc2cn(C3CN(C(=O)CCC(N)=O)C3)nn2)ccn1 N1(C(c2ccn(CC#N)n2)=O)CCC(NC(c2c(Cl)cccc2Cl)=O)CC(O)C1 C(=O)(C1=CS(=O)CCC1)NCCN(C)C(c1ccc(C(=O)CF)cc1)=O C1(C=C)(C(=O)NCC(CC=C)(C)CO)CCN(C(c2ncn(C)n2)=O)CC1 N1(C(C(C)n2ccnn2)=O)CC(C2CC2)(C(=O)NC2CC2C2CCCO2)C1 c1(OCC)cc(C(N2CCCC2)=O)c([N+](=O)[O-])cc1NCc1cnc(F)c(Cl)c1 C1(C)(CNC(CCC(CC)C)=O)COCCN(C(C2CCC(CC#N)CC2)=O)C1 N12CCCC(C1)OC(=O)C2c1nc(CC)sc1.C(=O)(C(C)C)NCCCC1CC1 N1(C(C=CSC)=O)CCCCC1C(=O)NC(C1CCN(c2ccncc2)CC1)C O=C(C1=CCCCO1)NC1CCCC(C(N2CC(CO)(CO)C2)=O)C1 c1(CCC)cccc(S(=O)(=O)Nc2c(C(C)C)cccc2C)c1 c1(NCc2c(C)ncn2C)[nH]c(=NC2CCCC(P(C)(C)=O)C2)nc2scnc12 C(=O)(C1CCCc2nccn21)NCC1N(C(c2c(C)cc(Cl)cc2)=O)CC(O)C1 c1(OC)ncc(C(=O)NCCCNC(C2(CF)CC2(F)F)=O)cc1F c1(C(C)C)nccc(C(=O)NC(c2ccccc2)CNC(C2CCCS2)=O)n1 N1(C(CN(CCC)C)=O)CCOCC1C(=O)NOCC(N1CCC(OC)C1C)=O Cc1cc(C)c(C)c(C(N2CCCC(C)(CNC(c3cc(F)n[nH]3)=O)C2)=O)c1C C1(C(=O)NC2CCC(NC(c3c(OC)cc(C)cc3)=O)C2)CN=C2N=CNN2C1 CC(CCC(=O)NCc1nccs1)NC(=O)Cn1ncn(C)c1=O c1(C(=O)OC)cc(C)nc(O)n1.c12cn(nn1)CC1(CC1)CNC(=O)NCC2 N1(C(COCC(=O)NOC2CCC2)=O)CC2CCC=CC12 CC1(C2(C(=O)NC(C3CCCCC3)C(=O)Nc3ccc(C4CC4)nc3)CC2)CC1 CCCCCCC(CC)NC(C1CCN(C(c2cc(CC)on2)=O)C12CCC2)=O C=CCC(C(=O)N(CC(C)N(C)C(c1cc(C(C)(F)F)n[nH]1)=O)C)C(C)C C1(C(=O)NC(C(C)NC(c2ccc(C(C)(C)C)[nH]2)=O)CO)CCC(F)(F)CC1 N1(C(C2CC3(CC3)CO2)=O)CCC2CC2(C(=O)NC2CC(O)CC2O)CC1 C(=O)(C(O)CC(N)=O)N1C(CNC(c2cccc(N(C)C)n2)=O)CC(O)C1 C12(CNC(C3(CC)CCCC3)=O)CN(C(=O)Cc3csc(S)n3)CC1CCO2 c1(SCCC)ccc(C(=O)NC(C2CN(C(c3cnco3)=O)C2)C)cc1 C(CCCCC(=O)N1CC2CC2(CNC(=O)CC2CCSCC2)C1)SC c1(CC)nc(C)[nH]c1C(N1CC(CCNC(C2(COC)CCOC2)=O)C1)=O CCC(C)CCC(=O)NC(C1(C(=O)NCC(C)CN2CCCC2)CC1)C C1(C(=O)N(C2CC2)CC2CCCN2C(C2CC(=C3CCC3)C2)=O)(OC)CCCC1 c1(OC)cc(C2CCCN2C(=O)NCC2(Br)CC2(F)F)ccc1O N1(C(CCN(C(CCC)C)C)=O)CCCCC(NC(C2CC(Cl)(Cl)C2)=O)C1 c1(OC)c(C)cc(-c2ncn(C)c2CN(CCCN2CCN(C)CC2)C)cc1C CCC(CC)C(=O)NCCN(C1CCCC1)C(c1cnn(CC2CCCO2)c1)=O C1(NC(C(C2CC2)OC)=O)COC2(C1)CN(C(=O)CCc1ccc(O)c(F)c1)C2 C1(CNC(CCSc2nc(C)[nH]n2)=O)COCCN1C(=O)CN1CC(C)(C)C1 c1(C(N2C(C(=O)Nc3nccc(Cl)c3OC)CC(=C)C2)=O)cc(C)cc(C#N)c1 N1(C(c2c(C)n(C)cc2)=O)CCN(C(=O)CN(C2CCC2)C)C(CC(C)(C)C)C1 CC1CC(CNC(c2csc(Cl)c2)=O)CN(C(c2ccc(O)cc2)=O)C1 CC1CCN(c2nnc(-c3ccccn3)n2CCS(=O)(=O)N(C)C)C1C C(=O)(C1=CC(C)(CC)C1)NC1C(CC(=O)NCc2nnc(CC)o2)C(O)C1 CC(C)(C)CC(O)C(=O)N1CCC(CNC(c2cc(O)ccc2Cl)=O)C1 C1(F)(C(N2CC(C)(OCC)C2)=O)CCN(C(=O)CC(C)CN(C)C)C1 C1(NC(C(c2ccc(CC)s2)=O)=O)CC(OC)CN(C(=O)CCCC(F)F)C1 CC1(C(N2CCOC(CC(=O)NCCC3CCCC3)C2)=O)CCCCC1 N1(C(Cn2ncc(CC)c2)=O)CCC(CCOC)(NC(=O)CS(=O)(=O)NC)C1 N1(C(C)=O)CC(O)CC1C(N1CC2CC1(CNC(C1CCC(C)(C)C1)=O)C2)=O C1(NC(C2(C)CC(=C)C2)=O)CCN(C(=O)C(C)N2CC(C)C2)CC(O)C1 C1(CNC(C(CN(C)C)(F)F)=O)C(C2CC2)CCN1C(=O)C1=CCCCCC1 C1(COC)(NC(=O)Cc2cc(Cl)n(C)n2)CCN(C(=O)C(F)(F)COC)C1 N1(CC(=O)NC(C(=O)NC2CC3CC3C2)c2cccs2)CC(=O)NC1=O C12CCCC(C1)NC(=O)C(C(C)=O)N2.c1(COCC)nc(CC)no1 C1(C(=O)Nc2c(C#N)scc2)Cc2ccccc2CN1Cc1ccc(O)c(I)c1 c1(C(N2CC(OC)C(NC(C34CCOC(C)(C3)C4)=O)C2)=O)cnc2c[nH]nc2c1 c1(C(N2CC(C)C(CCNC(c3[nH]nnc3C3CC3)=O)C2)=O)cc(Cl)ccc1O c1(C(CC)C)ccc(C(=O)NCCN2CCN(Cc3ccc(Cl)nc3)CC2)cc1 C#Cc1c[nH]nc1C(=O)NC12CC1CN(C(=O)CC1(c3ccccc3)CC1)C2 c1(NCc2c(C)nco2)ncnc(N2CCC=C(F)C2)c1C c1(C(=O)NCC2(c3ccc(Cl)cc3)CCCC2)cc(Cl)c(O)c(Br)c1 Cc1cc[nH]c1C(=O)NC(Cc1cnc[nH]1)C(=O)N1CCC(C(=O)N(C)C)C1 Cc1cnc2cc(C(N3CC(NC(c4cc5ccsc5s4)=O)C(O)C3)=O)ccn12 CC(c1cccs1)=CC(=O)N(C)CCN(CCOCCO)C(=O)C1CC1 N1(C(CC(C)C(F)F)=O)CCCC2(CCN(C(=O)C=C(C3CC3)C3CC3)C2)C1 C#CC1(C)CCN(C(=O)C(C(C)C)NC(=O)CCC2CCCO2)CC1 C1(NC(c2c(C)ccc(C(=O)OCC)c2)=O)CN(C(=O)CCSC)C2(CCC2)C1 N#Cc1cccnc1-c1cn(CCCCN2CCC(CN3CC=CC3)C2)nn1 C(C(C)NC(=O)Cc1cc(C)cs1)(C(C)C)NC(CN(C)CC)=O Cc1ccc(=O)n(CC(=O)NCC2(O)CCN(C(=O)C(C3CCCCC3)F)C2)c1 C1(c2cccs2)(C(N2CCC(NC(CC3(C)CC3)=O)C2)=O)CCCCC1 C(=O)(C#CC1CCOC1)N(CCCN(C(CC1CCN(C)C1)=O)C)C CC(C)CC(F)C(=O)NC1(CCCNC(=O)C(C)Sc2ccccn2)CC1 Cc1nn(C(F)F)cc1S(=O)(=O)N1CCC(NS(=O)(=O)C2CC2)C1 N1(C(CC2C(C)(C)OCC2)=O)CC2N(C(=O)CP(C)(C)=O)CCC2(C)C1 c1(C(=O)NC2CCN(C(C3CCC4CC34)=O)CC2)cccc([N+](=O)[O-])c1Cl C1(NC(C(CC=CC)C)=O)CN(C(=O)CN2CCSCC2)CC2CC12 N(C(=NCCCOc1ccccc1)NCc1ccccn1)Cc1n(C)cc(Cl)c1 C1(C(N2CCCC(CNC(=O)C=Cc3ccsc3)CC2)=O)CCc2nnnn2C1 C1(NC(COC(C)=O)=O)CC(CNC(C2CC2c2cccnc2)=O)CC1O c1(C(N2CCN(C(CC(C)(F)F)=O)C(C3CC3)C2)=O)cccc2c1CCO2 c1(C(N(CCNC(C(C2CCC(=O)N2C)C)=O)CC2CC2)=O)cnc2n1CCC2 C1(NC(C(CC)SC)=O)CC2CCC1N(C(c1ccns1)=O)C2 C(CSC)(C(=O)NCC1(CCNC(=O)COc2cc(C)on2)CC1)OC c1(OCC)cc(C(N2CCN(C(=O)COC(C)=O)CC2)C(=O)NC)cc(Cl)c1 C(=O)(CCCNC(=O)Cc1cscn1)N(CC=C)C1CC1 C12(C(=O)NC3C(C)CSC3)CC(CN1C(=O)CN1CCCC1)C2 C(=O)(CC(C)(C)C#N)N(C1CCC(NC(=O)CSc2ccccn2)CC1)C CC1(C)CCC(n2cc(CSCCNC(c3cc(O)nc(Br)c3)=O)nn2)CC1 C1(NC(C2Cc3nncn3C2)=O)CC12CCN(C(c1cnc(C(F)F)s1)=O)CC2 C12(CC(=O)N(CCC)C3CC3)CCC1CN(C(=O)COC(C)(C)CC)C2 N1(C(C(COCC)N=[N+]=[N-])=O)CCCC2CN(C(c3cccc(=O)n3C)=O)CC12 C=C(C)c1cccc(NC(C2CC2C(C)NC(=O)C(C)n2ccnn2)=O)c1 C1(C(=O)NCC(CNC(c2c(C)c(F)ccc2)=O)O)CC2(CCOCC2)CO1 c1(C(N2CCCC(n3cc(CCC(N)=O)nn3)C2)=O)cc2cc(Br)sc2s1 c1(CN2C(COC)CCOCC2)cnc2c(c1)CCC2 CC(C)CCCCCC(=O)N(C1CN(C(=O)Cc2cc[nH]n2)CC12CC2)C n1(CC)ccnc1C(C)NC(=O)C(C)=CCNC(C1(C)CC(C)C1)=O c1(OC)nccc(C(=O)NCC2(O)CCN(C(C3CC(C)C3)=O)C2)n1 c1(C(N(CC(C)NC(CN(CC)CC)=O)C)=O)ccc(CC2CCC2)cn1 N1(C(Cc2c(C)noc2)=O)CCC2(C1)CN(C(C1CC3CCCCC13)=O)CCO2 Cn1nccc1C=CC(=O)NCc1nocc1C(N1CCC1C(C)(C)O)=O N1(CC)CCOCC1C(=O)NCCC1CN(C(C2OCCOC2C)=O)C1 C1(C(=O)NCC2N(C(c3c(C(C)(C)C)noc3)=O)CCOC2)CC2CCC(C1)S2 c1(C(=O)NC2CCCC(NC(c3n(C)c(S)nc3)=O)C2)cccc(C2CC2)c1Cl C(=O)(CC(CNC(C1CCC1CC)=O)C1CCC1)N(CCCCOCC)C C#CC1(C(=O)NC(C)CCC2CC2)CN(C(=O)C(CC)CC)C1 C1(OC)CN(C(C2CC3CC3C2)=O)CC1NC(C1(O)CCCC1)=O N1(C(=O)NCC2CC(C)(C(C)(C)C)C2)CC2CC3(CCC3)C2C1 c1(C(=O)NCC2CCCCS2)coc(CNC(C2CC2(F)F)=O)n1 C1(CNC(C(C)CC(N)=O)=O)CC2(CO1)CN(C(C1CC(OC(F)(F)F)C1)=O)C2 S(=O)(=O)(c1c[nH]c2nc(Cl)ccc12)N1CCC(C)(CC(C)C)CC1 C1(C(N(C)CC2CCC(=O)N2)=O)CN(C(=O)Cc2ccns2)CC12CCC2 C1(CC)(NC(=O)C(N2CCNC2=O)C)CN(C(c2cc(C3(C)CC3)n[nH]2)=O)C1 c1(C(=O)NCC2CCN2C(=O)Cn2cnc([N+](=O)[O-])c2)cc2cccc(F)c2o1 Cc1ccoc1CC(=O)NCC(C)CN(C)C(c1csc(-c2cnccn2)n1)=O C1(NC(c2n[nH]c(CC)c2Cl)=O)CCC2CCN(C(=O)CC3CC3)C1C2 c1(COC)ccccc1C(=O)NCC12CC(CNC(C3C=CCCC3)=O)(CO1)C2 c1(N2CC(OCCNC(C(C3CCCC3)OC)=O)C2)snc(Cl)c1C#N c1(C(N(C2CCN(C(c3ccc(CO)s3)=O)C2)C)=O)ccn2cnnc2c1 C1(C(N(C)CC2(O)CCOC2)=O)CCN(C(=O)Cn2ccnn2)C1(C)C Cc1cncc(C(N2CCCC(NC(=O)CCn3cccn3)C2)=O)n1 Cc1cnn(CCC(=O)NC(C)CNC(=O)C=C2CCN(C)C2)c1 N1(C(C2CC(CCNC(C3CC(=C4CCC4)C3)=O)C2)=O)CCC2(CC1)CC2CO CC(C(CO)NC(C1CCOC1=O)=O)NC(C1(CC2CC2)CCC1)=O C(C(C(=O)NCc1cc(C(N)=O)no1)C(C)(C)C)NC(c1ccn(COC)n1)=O N1(CCC(=O)N(C)CC)CCC(Nc2ccc(SC)c(C)c2)C(C)C1 N1(C(c2c(C#N)scc2)=O)CCC2(CCCCC2NC(=O)CNC=O)C1 C(=O)(CC(C(F)(F)F)OC)NCCN(C(C(C(CC)O)C)=O)Cc1ccccc1 N1(C(C(C)CC2CC2)=O)CC2CC(C1)C2NC(c1ncsc1-c1ccccn1)=O C1(CC(N2CCC(NC(C3(N(C)C)CCOCC3)=O)C2)=O)OCCCC1(C)C Cc1ccc(C#N)c(N2CCCC(CNC(=O)Cc3nc(C4CC4)nn3C)C2)n1 c1(SCC(=O)NC(CNC(Cc2n(C)cnc2)=O)(C)CO)cccc(Cl)c1 N12CCCN(CC1)C(=O)c1ccccc1C2.c1(C(=O)OC)ccc(OC)s1 O(NS(=O)(=O)c1ccc(F)cc1)CC(=O)NC1(C)CN(C(C2(F)C(C)C2)=O)C1 N1(C(c2c(CC)nc[nH]2)=O)CCC(N=c2[nH]c3ncc(Cl)cc3o2)C(C)C1 C1(C)(C(=O)NC23CN(C(CN(C)S(N)(=O)=O)=O)C(CC2)C3)CC(C2CC2)=NO1 N1(C(c2cnc(C)[nH]2)=O)CC2(CNC(C3(O)CCC3)=O)CC2(C(F)(F)F)C1 c1(N2CCC(NC(Cc3ccc(C)c(C)c3)=O)C(C)C2)ncnc2c(C)csc12 c1(C(=O)NC2(CN(C)C(C3(F)CCOCC3)=O)CC2)cccc(F)c1N S(=O)(=O)(c1ccc2c(c1)NCC2)N1CCC(c2cc(C)no2)C1 C12(C(=O)OCC)CC(C)(CN1CC(c1cc(C)nn1C1CCOC1)=O)C2 c1(N2CCC(=C)C2)nc(N(CC(C)(CC)OC)C)c2c(n1)CSC2 Cc1c(C(N2CC(NC(=O)CSc3cccc(Cl)c3)C(C)C2)=O)ccn1C CC(C)C(C)(C)C(=O)NCC1C(O)C(O)CN1C(=O)C=CS(C)=O C(=O)(C1CCc2sc(NC(=O)CC3CC3NC(=O)OC(C)(C)C)nc21)OCC N1(C(C=C(C)C(C)(C)C)=O)CCCC(N(C)C(C2(O)CC2)=O)CC1 CCC(CC)CC(=O)N1CCN(C)C(CNC(=O)C(C(F)(F)F)OC)C1 c1(C(C(=O)NCCC(C)NC(c2cccnc2F)=O)(C)C)cccc(Cl)c1Cl CC1(C)C(NC(=O)COC2(C)CCCC2)CCN1C(=O)CC1CC2C=CC1CC2 C1(NC(C2(SC)CC2)=O)CCCC(N(C)C(c2ccc(CCCO)cc2)=O)C1 C=C(Cl)C(C)(C)C(=O)NC1COCCN(C(c2cnc(C(C)O)s2)=O)C1 C1(C(=O)NCC2(C(N(CCCOC)C)=O)CCCO2)CN(C)C(=O)N1 N1(C(c2cc(C(F)(F)F)c[nH]2)=O)CC(CNC(C23COCC2C3)=O)C(O)C1 c1(SCC(=O)NC2(CNC(Cn3ccc(C)n3)=O)CCC2)nc2ccccc2o1 N1(C(C(C=C)O)=O)CC2CCCC(NC(=O)CC3CCCCC3C)C2C1 C1(C)(COC)CN(C(=O)C(C)(c2cccs2)NC(=O)CC(SC)SC)C1 C(=O)(C(O)(C(C)C)C(F)(F)F)N1CCCC(O)(CNC(Cc2cnc(C)[nH]2)=O)C1 C1(C(=O)NCC2C(NC(c3ccc(CC)[nH]3)=O)CCC2)CCC(=O)N(C)C1 C1(NC(CCC(CC)C)=O)CCC12CCN(C(C1CC1(Cl)C(=O)OC)=O)CC2 N1(C(C=CCNC(c2c(C)[nH]cc2)=O)=O)CCC(C(C)CO)CC1 Cc1c(C(N2CCC3CCN(C(c4cccn4C)=O)CC23)=O)sc2ccccc12 C1(C(N2CCCC(CNC(CC(CC)O)=O)C2)=O)CCc2nncn2CC1 C(C(C)(F)C(C)C)NC(CN(C(=O)C(CCOC)OC)CC)=O C(=O)(C1CCc2c[nH]nc21)NCc1occ(C(N(CCNC(N)=O)C2CC2)=O)c1 CCC(C(C)CN(C)C)NC(=O)C(C)NC(c1cncc(NC)c1)=O C(c1cncc(F)c1)=CC(=O)NC1CC(CNC(C2CC(OC)C2)=O)CC1O C1(CC(=O)NC(C(N2C(C)(C(=O)NC)CC2)=O)Cn2cccn2)CCC(C)CC1 C1(NC(C2C(CCC)C2)=O)CC12CCN(C(c1cnn(C(C)C)c1)=O)C2 c1(C(=O)NC23CC(C(=O)NCC4C(C)(C)CCC4)(C2)C3)cc(N)cc(F)c1 Cc1cc(CNC(C2CCN(C(=O)Cn3cnnc3O)C2C(C)C)=O)cc(O)c1 Cc1cccc(C)c1OCCCN1CCCC(C(N2CC(C)CC(C)C2)=O)CC1 C1(C(=O)NC2C(C)CCN(C(C3(O)CCSCC3)=O)C2)CCC2C(CC1)C2(F)F N1(C(C(c2ccccc2)C)=O)CC(CNC(=O)C=Cc2ccncc2)C(C)C1 c1(C(=O)NC2CC(C)N(C(C3CC(=C4CCC4)C3)=O)CC2)c(Cl)cc(Cl)cc1Cl C1(CNC(C(C=CC)O)=O)CCCN(C(=O)Cc2csc3nccn23)CC1 c1(C(=O)NC2CN(C(=O)C(O)c3ccsc3)C2)csc2cccc(F)c12 C=CC(F)(F)C(=O)N1CC2CC1C2C(=O)NC(CCO)C1CC1 N1(C(c2c(C)nc(COC)s2)=O)CCN(C(=O)C2=CCSC2)CC1c1cn[nH]c1 c1(C(N(CC(CC)NC(C2(N(C)C)CCOCC2)=O)CC)=O)cccc2ncnn12 C1(C)(CNC(C(C)NC(C(c2ccn(C)c2)C)=O)=O)CCC2(CC1)CC2 c1(C(=O)NCCNC(CCOCC#C)=O)cc(Cl)c2c(c1)OCCCO2 C1(O)(CNC(C2CNC(=O)O2)=O)CCN(C(c2cc(C(F)F)on2)=O)CC1 CCC(C)CC(=O)N1CCOCC1CCNC(=O)C(=Cc1c[nH]cn1)F N1(C(C(CC)OC)=O)CC2(CC(NC(C3(COC)CCCCO3)=O)C2)C1 C12(NC(c3cn(C)nc3)=O)CC3CCC(C1C2)N3C(c1cnc(N)c(CO)c1)=O N#CC1CCCCC1NC(=O)C(CC1CCC1)NC(=O)CCCN1CCCC1 C1(NC(c2cn(C)nc2C(C)(C)C)=O)COC2(C1)CN(C(=O)C(C)(C)C(N)=O)C2 CC1CN(C(c2ccoc2CNC(C2COC(=O)N2C)=O)=O)CCO1 C1(C)(CNC(COCCC)=O)CCCN1C(c1cn(C)nc1SC)=O CCC(C)(O)C(=O)N(C)CC1(NC(c2ccc(Cn3cccc3)cc2)=O)CC1 C(=O)(C(O)C(F)(F)F)N1CCCC(CC(=O)NC(C23CCC(CC2)C3)C)C1 C1(C(N2CCC(C(=O)NCCN3CCCC3CO)C23CC3)=O)CC2CCCC2C1 C1(NC(COCCOC)=O)CCCC1(C)CNC(C1CCCN1C(C)=O)=O N1(CC(=O)NC2C(C)(C)C2)C(=O)c2cc(Cl)c(Cl)cc2C1=O N1(C(C(=Cc2cccs2)C)=O)CC(NC(=O)C=Cc2cn[nH]c2)C2CC12 c1(C(=O)NCC2CC(O)CN2C(C2C=CC=CC=C2)=O)cc(Cl)ccc1[N+](=O)[O-] CCC(C)CC(C(=O)NOCc1nc[nH]n1)NC(=O)C=Cc1cocn1 n1(CCC(N2CC(CC=C)(NC(=O)CC(C)(F)F)C2)=O)cnc2sccc2c1=O C1(CNC(CC2N(C(c3ccc(C(N)=O)[nH]3)=O)CC2)=O)OCC2CCC1C2 c1(C2C(CN3C(CN(C)C)CCC3)C2)ccc(F)c(F)c1.C12CCCN1C2=O C1(NC(C=CC2(C)CCOCC2)=O)CCC2(CCN(C(C3CCOC3)=O)CC2)C1 Cc1c(C(=O)N(C2CN(C(=O)Cn3cccc3)CC2(C)C)C)ccc(F)c1F CC1C2CCC(C2)C1C(=O)NCCn1ccc(C(N2CC(C3(C)CC3)C2)=O)c1 C12(NC(c3nc(C)sc3)=O)CCCC1N(C(C1(C(F)(F)F)CC=CC1)=O)CC2 N1(C(c2c(C)c(Br)c(Br)s2)=O)CC2CC(CC(=O)O)C(C2)C1 CCC(O)C(=O)NCC1CCC1.C(=O)(CCNC(=O)OC)N1CCC1 C(C(C(=O)NCCCN(C1CCCC1)C(=O)C=CC=C(Cl)Cl)OC)OC c1(OCC(=O)N(CCC(C)NC(c2ccc(CC)o2)=O)C)c(C)occc1=O C1(NC(C(C)=C2CCC2)=O)CC1C1CCN(C(c2ccnc(C)c2N)=O)CC1 C(CCC(C)C(=O)NCCCN(C)C(c1cccc(OCC(F)(F)F)c1)=O)OC C1(NC(C2(COCC)CC2)=O)CN(C(=O)C=Cc2cn(C)cn2)CC1C(F)F N1(C(C(C)OCCCC)=O)CC2CCN(C(c3nccc4ccsc34)=O)C2C1 c1(CC)cc(C(=O)Nc2c(CC(C)OC)cccc2)cc(C(=O)O)c1 c1(N(C2CCC2)Cc2c(C)cccc2)cncc(S(C)(=O)=O)n1 c1(C(N(CCC(C)NC(C(CC)C2CCOCC2)=O)C)=O)ccccc1Cl NS(=O)(=O)c1c(Nc2cc(NCC3C4CCCCC34)ncn2)cc(F)cc1F Cc1nn(C)c(=O)c(C(=O)NC2CN(C(=O)C3=NOCC3)CC2O)c1C Cc1cccc2nc(C(=O)NC3(CO)CCCN(C(=O)C4=CC(C)(C)C4)C3)cn12 C1(C(N2CC3C(CNC(COCC(=O)NC)=O)(C3)C2)=O)COC2(CCC2)C1 C(=O)(CCS(C)=O)N1C(CNC(COCc2ncc(C)o2)=O)CC1 CN1CC(C)(C(N2CCCOC(CNC(c3cscc3C(F)F)=O)C2)=O)CC1=O c1(N2CCN(C(CCC(C(C)C)C)=O)CC(O)C2)nc(Cl)nc2c1ncn2C C(=O)(C(C(C)(C)C)NC(=O)CC1CCC=CCC1)N(CC=C)CCOC c1(C(N2CCCC(N(C(=O)CCCCF)C)CC2)=O)cc(Cl)cc(F)c1N C1(CC(=O)NC(=O)NCCCCC2CC2)(CO)CCOCC1.c1ncc[nH]1 N1(C(c2cnc(=N)[nH]c2)=O)CCC(C2CCN(C(=O)Cc3ccns3)CC2)C1 c1(C(=O)NCC2CN(C(CCC=CCC=C)=O)CC2C)c(F)cc(C#C)cc1F N1(C(CCOCCOC)=O)CCCCC(C(=O)Nc2cc(OC)nc(C)n2)C1 N1(C(CSCCOC)=O)CCCCC1CCC(=O)NC1(C)CS(=O)(=O)C1 C1(C(NOC(C)C)=O)CC2(C1)CN(C(c1cc(F)c[nH]1)=O)C2 C1(CC(=O)N(CC(CNC(C(CC)OC)=O)C)C)CCC2(CC1)CC2 C1(CC)(CC)CC(NC(=O)Cc2cnoc2)CN1C(=O)CC1CCC(O)C1 C1(C2CCN(C(C3CCCCC3)=O)C2)(NC(Cc2ccn(C)n2)=O)CC1 C(C(=O)NCC(CO)NC(=O)Cc1ccccc1OC(F)(F)F)(C(C)C)SCC Cc1c(C(=O)NCC(O)CNC(C2(C(C)(C)O)CCC2)=O)ccn1CCO N1(C(c2ccc(CCC)[nH]2)=O)CCN(C(=O)C(C)(C#N)CC)C(C)C1 C(CN=c1ccc(S(=O)(=O)N2CCC(CCC)(CO)C2)c[nH]1)N(C(CC)C)C CC1(C(N2CCC(NC(c3ccc(C#N)o3)=O)CC2)=O)CCOCC1 N1(C(c2c(C)c(Br)n(C)n2)=O)CC2(CCCC2NC(c2ccn(C)n2)=O)C1 c1(C(N2CC(O)(C(C)NC(C(CC)F)=O)C2)=O)cnn(C)c1C c1(CNC(C(C)OC)=O)cc2n(n1)CCN(C(C13CCC(CC1)C3)=O)C2 Cn1cnc2cc(C(N3CCC(OCCNC(C4CSCCS4)=O)C3)=O)cnc12 C1(CC=C)(NC(c2nn(C)cc2SC)=O)CCCN(C(c2ccnnc2C)=O)C1 C1(NC(CN(C)C)=O)CN(C(=O)C(F)CC2CCCCC2)CCC12CCC2 c1(NC)cc(Cl)ccc1C(=O)NCCCNC(=O)COCC1CCCO1 C=CCCCC(C(=O)NC)N1CCC(OCC(=O)OC)C1 C(=O)(C(C(=O)N(CC(C)NC(C1CCN(C(C)C)CC1)=O)C)C1CC1)OCC CN(CP(C)(C)=O)CC(C1CC(C)(C)C1)O N1(C(C(CC)(C)C)=O)CCCN(CCNC(=O)C(F)(F)COC)CC1 C1(NC(C2C(OC)C2)=O)CCOC12CCN(C(=O)Cn1nc(C)oc1=O)CC2 CCC(C)C(O)C(C)C(=O)NC(C)(C)CC(F)C(=O)NCC1CC2C=CC1CC2 C1(NC(=O)C(F)n2cccn2)CN(C(C2(CF)CC3(CCC3)C2)=O)CC12CCC2 C(C)(C)(CCC(=O)NC1CC(C)N(C(=O)CC2(C)CCC2)C1)OC N1(C(C(C)OC)=O)CCC2(CC1)CCN(C(=O)CN1CCCCC(O)C1=O)C2 C(N=c1[nH]c(=NCC(C)(C)c2ccccn2)[nH]c2c1SCC2)c1c(C)cn(C)n1 Clc1cccc(Cl)c1N1CCN(CC2CCCC23CC3)CC1 C(CCC(C)C(=O)NC1CC1NC(c1cccnc1NC(C)=O)=O)OC N1(c2nc(SC)nc(Cl)c2)C2CCC1CC(NC(=O)CC1OCCC1C)C2 c1(C(=O)NCC(C)(O)CNC(c2c(CC)cco2)=O)oc(CO)nc1C c1(NC(CC)CCOC)ccc(S(=O)(=O)NCC2CC23CCC3)cc1Cl N1(C(c2nc(NC(C3CC3C3CC3)=O)sc2)=O)CCc2cc(F)ccc2C1 c1(C(=O)NCCN(C(C2CC(C(C)C)C2)=O)C(C)C)ccncc1 N1(C(C(C)OC)=O)CC(CC(=O)NCC2CCCC(CO)C2)C2(CC2)C1 CC1CC(NC(=O)CCC2(C)CN(C(c3ncccc3O)=O)C2)CCN1C C(S(=O)CC(=O)N(c1ccc(Oc2ccccc2)cn1)C1CC1)c1[nH]cc(C)c1 n1(C(C)C)cnc(C(=O)NCC2CCC2NC(c2ccsc2-n2cnnn2)=O)c1 C(=O)(C1=CC2(CCOC2)C1)N1CC(CC(=O)N(C(C=C)C)C)C2(C1)CC2 N1(C(c2cc3cccc(Cl)c3o2)C(=O)NCCCC)CC=CCC12CCCCC2 C(CC(C)NC(c1ccoc1)=O)NC(=O)CO.C(=O)(CC1CC1)NCC C1(C(=O)NCC2C3CN(C(C4C(OC(C)(C)C)C4)=O)C2C3)CC2(CCCC2)CO1 c1(C(=O)NC23CC(C2)N(C(C2CCC(F)(F)C2)=O)C3)ccc2nonc2c1 CCCCC(O)CC(=O)NCCCC(C)NC(=O)Cc1ccn(C(C)C)n1 c1(C(c2n(CCC)nnn2)NCCC2COC2)ccc(S(=O)(=O)N(C)C)cc1 c1(-c2cccc(C)c2F)ccc2c(C(N3CCn4nccc4C3)=O)cnn2c1 c1(C(N(C2CCN(C(c3cc(Cl)c[nH]3)=O)CC2)C)=O)ccc(F)c(F)c1N C1(N(C(CN(CC)CC)=O)CCO)CCCN(C(=O)Cn2nccc2C)C1 N1(C(C2(C)C(CC)CCC2)=O)CCCC2(NC(C3CCCC3(F)F)=O)CC2C1 C(C(C)CC(=O)NCc1nnn(C)c1C)NC(c1n(CCC)ncc1)=O N1(C(CCCN(C(=O)OC)C)=O)CCN(C(C2CCCCCC2)=O)C(C)CC1C C(=O)(C(C)(C)C(C)C)NCCC(=O)N(CC(=O)NCCOC)C C(CC(=O)N1CC2CC(OC)C(C2)C1)(C(C)(C)C)NC(C(CC#C)O)=O CC1CCN(C(=O)C=Cc2cscn2)CC1NC(c1cc(C2(C)COC2)no1)=O c1(-c2cc(CC(N3CC4COCC4C3)=O)ncc2)ccc(OC)c(F)c1 C(=O)(C(C)(O)C(F)(F)F)N1CCC(=C(C)C)C1.C1CN1 Cc1nc(C(=O)NC2(CNC(=O)CC3CC3(Cl)Cl)CCC2)cn1C c1(C(=O)NCC2N(C(c3ccc(C(=O)OC)s3)=O)CC=C2)ccnc(C)c1 N1(c2ncc(C)cn2)CC(NC(c2cccc3cccnc23)=O)C2CCCCC12 c1(CC(C)NC(CN(C(=O)CCCc2cnn[nH]2)C(C)C)=O)cnn(C)c1 N1(C(Cc2n(C)ncc2)=O)CCC(C(N2CCC(CCO)C2)=O)(CO)C1 c1(CNC(=O)C(=O)Nc2ccc(-c3ccc(Cl)cc3)s2)cnc(-n2cncn2)nc1 C1(OCP(C)(C)=O)CCCN(c2ccccc2OCC2CCCO2)C1=O c1(C(N2CC(CCNC(=O)C#CC3CC3)(OC)C2)=O)c[nH]c2cc(F)ccc12 CCS(=O)(=O)c1nnc(CCN(C)CCO)n1C1CC1.C(CC(N)=O)S N1(C(CC2N(C(=O)OC(C)(C)C)CSC2)=O)CCCC1(C)C1CC1 c1(C(=O)NC2CC(NC(C(C)NS(C)(=O)=O)=O)C(O)C2)cc(O)cc(C#N)c1 c1(OC)ccc2nc(C(N3CC(NC(=O)C(C)(C)SC)CC3(C)C)=O)ccc2c1 CC(F)(F)C(F)C(=O)NC1C2CC3C(C2)C13C(=O)NCCn1ncccc1=O c1(C(=O)NCCCN(C(C2C(C)(CC)C2)=O)C)cc(C)nn1-c1ccccc1 C1(CNC(c2cnn(C)c2F)=O)COCCN(C(=O)CCN2CCNC(=O)C2)C1 N#CC1(C(N2CC3(C2)CN(C(=O)C=CC2CCC2)C3)=O)CC2CCC1C2 c1(C(N(c2ncccc2N)C)=O)cc(-c2ccc(F)nc2F)c2n[nH]cc2c1 C(CC(O)C(=O)NN1C(=O)CCC1C(=O)Nc1ccc(Br)cc1)NC(C)=O C1(O)(C(C(=O)NC2C(NC(CC3CC(C(=O)OC)C3)=O)C2)F)CCCC1 c1(C(=O)NC(C2CCN(C(C3N(C)CC(F)C3)=O)C2)(C)C)cnc2ccoc2c1 c1(C(N(C2CCN(C(=O)CC3CCC3(C)C)CC2)CC)=O)cc(F)c(O)c(Cl)c1 C1(NC(CC2C(NC(C(C)N3CCCC3)=O)CCC2)=O)CC2(CCC2)C1O c1(C(=O)NC(CNC(=O)C(F)(F)c2ccncc2)C2CC2)ccncc1Cl C1(O)(C(C(=O)NCC2CCN(C(C3(CC#C)CCOC3)=O)C2)(F)F)CCOCC1 C1(C(=O)NCC2(O)CCN(C(C=CC(CC)=CC)=O)C2)CCc2nc[nH]c2C1 c1(NC(C2CCCC2NCc2cnc(Cl)cc2Br)=O)ncc(Br)nc1Cl N1(C(c2cc(S(C)(=O)=O)sc2)=O)C2CCC1CN(C(=O)CC1CNC(=O)C1)CC2 C1(NC(C(C)SCCCC)=O)CCC(CCNC(c2sccc2COC)=O)C1 C1(CNC(C2=CC(C)C2)=O)CCCCN(C(=O)Cn2nccn2)C1 c1(CN2C(CNC(c3ccc([N+](=O)[O-])o3)=O)CCC2)c(F)cccc1Br c1(C(N2CCC(C(C)C)(C(=O)NC(C)Cn3cncn3)C2)=O)cnccc1C#N C1(CC(=O)N(C2CCCC2C#N)C)C2CCCC2N1C(c1ccncc1Cl)=O C1(CNC(c2cnc(C3CC3)o2)=O)CN(C(=O)CC2=CCCCC2)C2CCN1C2 C1(CCC)CN(c2ccnc(COC)n2)CC1N(C)C N1(C(C(CSCC)NC(CCC(=O)NCC)=O)=O)CC2(CCC(=O)N2)C1 N12CCCC1C1CCCN1C(c1cc(C)ns1)C2=O.C1(CNC(C)=O)CCCO1 C12(C(N3CCCC(C(C)(C)O)C3)=O)CCC(C)(C1)OC2.C12(CCCCC1)C(=O)N2 c1(C(=O)NCCNC(C(CC(=C)C)NC(C)=O)=O)oc2ccc(Cl)cc2c1C c1(C(N2CCC(C)(CNC(C3(F)CCOC3)=O)C2)=O)cc(F)c(F)c(C#N)c1F c1(C(=O)NC(C(C)C)CNC(c2cccn2C)=O)c(F)cncc1Cl C1(O)(C(C)CNC(=O)C2CC2)CCN(C(c2ccc(C(N)=O)o2)=O)C1 c1(SCc2nnc(-c3c(C)n(C)nn3)n2C2CCCC2)cn2c(n1)CC(C)CC2 N1(C(CCSCCC)=O)CCC(C)C(CNC(c2cnc(C(N)=O)s2)=O)C1 CCCCCC(C)CC(=O)NC1CN(C(=O)Cc2c[nH]nc2C)CCC1O c1(C(=O)NCCCC(C(=O)N2CC(C(CC)C)C2)O)ccc2n[nH]cc2c1 Cc1nc(O)c(C(=O)N(C)CC2CCN(C(c3cc(F)c[nH]3)=O)C2)cc1Br C1(CC)C(NC(=O)CCC2CC2CC2CC2)CCN1C(c1cccc(Cl)c1)=O c1(C(=O)NC2CCCCN(C(C3CC(C)(CC)C3)=O)C2)ccc2c(c1)C=CCC2 c1(SCC=C)ccccc1C(=O)NC1CC(C)N(C(=O)CCCc2cc[nH]n2)C1 c1(C(=O)NC(CNC(C(CCC)OC)=O)C)cc(F)cc2nc[nH]c12 C1(NC(Cc2cccc(SCC)c2)=O)CC2CCC1(NC(c1cn(C)cn1)=O)C2 Cc1c(C(=O)NC2CC(O)CN(C(=O)CCC3CCC3)C2)sc2ccc(F)cc12 c1(OC)cc(NC(c2cn(C3C4CC5C(C4)C35)nn2)C(C)C)cnc1Cl CC(C)C(F)(CNC(c1cccc(C2CC2)c1)=O)C(=O)NC1CCCN(C)CC1 Cc1nc2c(cnn2C(C)C)cc1C(=O)NCCC(C)CCNC(=O)C(C)C#N CC1C(CC(=O)NCCOCC(N2CCC(CC3CC3)C2)=O)C1(F)F C12(C(N(CCCNC(C(N3CCC(C)CC3)=O)=O)C)=O)CCC(C#N)(CC1)CC2 C(=O)(C(C#N)CC)NCC1(CCNC(C(C=C)O)=O)CC1 Cc1cc(C(C)C)nc(=NCC(C)CNC(c2cccc(C(N)=O)c2F)=O)[nH]1 Cn1ccc(C(N2CC(O)(CNC(=O)CC3CCN(CC(F)(F)F)C3)C2)=O)c1 C(=O)(C(CO)C(C)(C)C)N(CCN(C)C(c1cn(C)nc1C(F)F)=O)C c1(NC(C)=O)cc([N+](=O)[O-])c(Cl)cc1C(=O)NC1CC(C)(NC(C2CCC2)=O)C1 N1(C(C(CC)(C)O)=O)C2CCC1CC(NC(c1cccc(=O)n1O)=O)C2 Cc1cc(F)c(Br)cc1C(=O)NCC1CCC(C)CN1C(=O)CC(F)F c1(OCC(=O)N(CCN(C(C(C2CCC2)OCC)=O)C)C)cc(C)cc(C)c1 Cc1ccc(C(N2CC(CC(F)C(=O)N(CC(N3CCCC3)C)C)C2)=O)cn1 C(CN=C(NC1CC1)N(C)Cc1cnc(C(C)CC)nc1)n1c(C)ncc1 c1(C(=O)NCCOCCNC(c2c(C)cc(SC)o2)=O)c(C)nc2ccccn12 c1(C(=O)NCC2(F)CCN(C(C(C(=O)OCC)OC)=O)C2)cnc2n1CCOC2 c1(C(N2CC(C)CC(NC(COC)=O)C2)=O)cc2c(Br)coc2cn1 C(C(C)(C)CNC(=O)CC(O)c1ccccc1)N(C(=O)COCC1CCCC1)C c1(OC)cc(O)c(CN2CC(C)(C(=O)NC(C)CN(C)C)C2)cc1Br C(C)(c1ccccc1)=CC(N1CCC(OCCNC(C2C(CCC)C2)=O)C1)=O C(=O)(C(O)C1=CCCCC1)N1C(CNC(c2n(CC)nc(C)c2)=O)CN(C)CC1 C1(n2cc(C(C)O)nn2)CCCN(C(=O)COc2ccc(Br)nc2)CC1 c1(C(=O)NCC2(CC3(C(N(C)C4CC4)=O)CC3)CC2)ccc(C(F)(F)F)cn1 c1(C(=O)NCC2CCN(C(CCOc3c(C)cccc3)=O)C2)c(Cl)nn(C)c1Cl N1(C(C2(C#C)CC2)=O)CC2CC(C1)CN(C(c1coc3c1CCCC3)=O)C2 N1(C(CCC)=O)CCCC1C(=O)N(C(C)CN(C)C(c1cscc1Cl)=O)C N1(C(C2COC(=O)O2)=O)CCOCC(NC(C2CN(C(=O)OC(C)(C)C)C2)=O)C1 N1(C(CCc2cc(C)no2)=O)C2CCC1CN(C(=O)C1=CCCCO1)CC2 C1(C(=O)NCC#CC(=O)NCC2(F)CCOC2)(CC)CCCC1 C(C(COC)C(=O)N(C(c1ccccc1)CNC(C1C2CCCC12)=O)C)OC C1(Cn2cc(CCN(C(C)(C)C)C)nn2)CCCCN1C(c1ccc(O)cc1)=O CC(N=[N+]=[N-])C(=O)NC(CCC1CCC1)C(=O)NCc1cccc(O)n1 C1(NC(C(C)CC2CCCCC2)=O)CN(C(c2nnn(C)n2)=O)CC1(C)C N1(C(=O)NCc2c(C)n(C)nn2)CCC(=C(F)F)CC1 c1(SCCC(N2CC(NC(C(c3ccccc3)SC)=O)C2)=O)ccccn1 c1(OC)ccncc1C(=O)NC1CCC(NC(C2(Oc3ccccc3)CC2)=O)C1 CC(C)C(O)CC(=O)N(CC(C)NC(=O)C(C)CSc1ccccc1)C C1(C(=O)NCC2(Cc3ccc(O)cc3)CCC2)CC2CC1N(CC1CC1)C2 C1(C(N(C)CC2(CNC(C(C=CC)O)=O)CC2)=O)CCS(=O)(=O)C1 [N-]=[N+]=NCC(O)CN1CCN(C2CCCCC2O)CC1 CCC(C)C(C(=O)N1CCOCC1CCNC(C12CC(C)(CO1)C2)=O)NC(C)=O c1(CC(C)C(=O)N(CC(O)CNC(C2(c3cc[nH]n3)CC2)=O)C)ccc(Cl)cc1 C(CCC[Si](C)(C)C)N(CCN(C(c1ncc(Br)cc1C)C(=O)NC)CC)C c1(C(=O)NC(C2CN(C(=O)C3=CCC3)CCO2)C)cc2c(F)c(Cl)ccc2[nH]1 C(CCCC(C)NC(=O)C(C)CN1CCCCC1)NC(C1(CCCC)CC1)=O c1(CN(CC(=C)C)C(c2ccc(CN3CCOCC3)s2)=O)ccc(SC)cc1 C1(NC(C2N(C(CC3(CSC)CC3)=O)CC(F)(F)C2)=O)CC=C(C(C)C)CC1 C1(NC(c2cc(C(C)=O)sc2)=O)CCCCCN(C(c2cc(C)c(C)[nH]2)=O)C1 N1(C(CCc2nnc(C)n2C)=O)CCC2CN(C(=O)C(c3ccc(Cl)s3)C)CC12 n1(CC)cc2ccc(C(=O)NCC3(CNC(=O)C(CC)OC)CCC3)cc2n1 c1(OC)ccc(F)c(C(=O)N(CCCN(C)C(C2(C)CC2Br)=O)C)c1 N1(C(c2cnn(C)c2Cl)=O)CCc2cc(-c3cccc(CCO)c3)ccc2C1 Cc1cc(S(N)(=O)=O)sc1C(N1CC2CCC(C1)N2C(C1(CO)CC1(F)F)=O)=O c1(CNC(C2CCN2C(=O)C(c2cccc(Br)c2)O)=O)cc(Br)cc(Br)c1 C#CCC(O)C(=O)NC(C1(O)CN(C(=O)C(C)(C)C2CCCC2)C1)C C1(C(N2C(CN(C(c3nnc(CC)s3)=O)C3CC3)CCC2)=O)OCCOC1(C)C CCC(C(=O)NCCCCC1(NC(=O)Cc2nc(C)sc2C)CC1)C(F)(F)F N1(C(C2(CC#C)CCCCC2)=O)CCN(C(=O)Cc2ccccc2C)C(CC)C1 c1(C(N2CCCC(NC(CNC(CC)=O)=O)C2C)=O)ccc2c(c1)CC(=O)N2 N1(CC(N2CC(C)N(C(=O)C#CC3(C)CC3)CC2C)=O)CCCC2(CC2)S1(=O)=O N1(C(C(C=C)(C)CC)=O)CC2CCC1CN2C(=O)C=Cc1csnc1C N1(C(=O)C=CC2CCOC2)CCCC(CNC(C2(Cl)CC2)=O)C1 Cc1cc(C(=O)NCCNC(c2sccc2C(C)C)=O)cn1C c1(COC)nc(NCCc2cccc(SC)c2)cc(N2CC3CC2C3)n1 N1(CC(=O)NC(COC)C)CCN(C(=O)CC(C)n2ccnc2)CC1 c1(CNC(C(C)CC(F)F)=O)cccc2c1CN(C(C1CC1C1CC1)=O)C2 c12ccc(cc1)NC(=O)N2.C1(C(C)C)C(CNC(=O)C2CC2)C1(F)F.C1CO1 c1(CC)ccc(C=CC(N2CCCC2(C)CNC(c2cc(C(C)=O)c[nH]2)=O)=O)o1 CCCC(C(=O)NC1CCCN(C(c2cc(F)cc(F)c2F)=O)C1)C(C)C C1(C(=O)OCC)CC2(CCN(C(=O)C=CC=C(Cl)Cl)CC2)CN1C(C)=O C(=O)(CS(=O)(=O)c1ccccc1)NC1CC2CN(C(c3cc(CC)on3)=O)C1C2 N1(C(c2cc(COC)oc2C)=O)C2CCC1CN(C(=O)CCOCC(C)C)C2 c1(CC)cccc2c1OCCC2Nc1cc(Br)c(O)cc1Cl N1(c2cc(N3CC(CC)N(CC)CC3)ncn2)CCC2(CC1)C(=O)NCCN2C Cc1sc(O)nc1C(N1CC(=C(F)CNC(C2CC2c2ccccc2)=O)C1)=O CC1(C)CCN(C(=O)C(=O)NC2CC2)CC1CNC(=O)CC1(CO)CCCCC1 C1(CC)CN(C(c2ccc(OC)s2)=O)CCN1C(c1cccc(OC)c1)=O c1(C(c2n(CC=C)nnn2)NCc2nc(C)ns2)nc(F)ccc1Br C(=O)(C(O)CC(F)(F)F)N1C(CCNC(=O)CN2CCCCC2)CCCC1 C1(C)(C(N(C)CC2(O)CN(C(c3c(C)c[nH]n3)=O)C2)=O)CCCN1C CC(C)C(F)(F)CC(=O)NC(C)C(C)NC(c1cc(Br)c(O)cc1F)=O C1(C(N2CCC(O)(Cn3cc(C(C(C)C)O)nn3)C2)=O)CC2OC(=O)OC2C1 CC1C(C(N2CC(CO)C2(C)C)=O)CCN1C(=O)COc1ccn(C)n1 Cc1[nH]c(C)c(C(N2CCC2(C)C(=O)NCC(=O)NC2CC2)=O)c1C C1(C(N2C(C3(C)CC3)CCCC2)=O)CCN(C(=O)Cn2ccnn2)O1 C12(C(N(CC(C(=O)OC)C)C)=O)CC1CN(C(=O)CC1CCC(C)(C)C1)C2 CCCCC(CC(=O)N1CCC(CF)CC1)NC(=O)CCC1CCCO1 N1(CC)N=C(C(=O)N(C)CCOCCN(C(=O)CC(CC)C(F)F)C)CCC1=O CC1CC(=O)NCC1C(=O)NC(C)(C)CN1CCN(C(=O)C2=CCC2)CC1 C1(C(=O)NC(CC(=O)OC)C2CC2)CC12CN(C(=O)COc1ccccc1C)C2 C1(NC(c2ccc(CO)o2)=O)CN(C(C2CC3C=CC2O3)=O)CC2CC12 C1(C(=O)NC2C3CCC2CC3)CN(CC2COCCO2)CCC1O N1(c2nnc(C)o2)CCC2(CCCC2NC(c2cccnn2)=O)CC1 C1(C)(NC(c2ccc(C)nc2)=O)CCCN(C(=O)CCCc2ncco2)C1 C(=O)(C(CO)C(C)(C)C)N1C(CC(=O)NC(CC)Cn2cncn2)C2CCCC21 C1(C(=O)NC2C=CC(CC(NOCC=C)=O)C2)CCC2(CC1)CC2 CCCCCCC(=O)NCC1CC(C(N2CC(N3CCCCC3)C2)=O)CO1 C1(NC(CCC=C)=O)CCC(COC)CC1.C12CC(C1)C(=O)N2 Cn1nnc2c1CCN(C(=O)C(C(C)(C)C)NC(C1CCCOCC1)=O)C2 Cc1nc(=NC(C)c2c(F)ccc3ccccc23)[nH]c2ccccc12 C1(CC)C(=O)NCCN1C(=O)C(CN=[N+]=[N-])NC(c1cnc(C)o1)=O c1(C(C(=O)NCCN(C(C(CC)OCC)=O)C(C)C)(C)O)ccc(Cl)cc1 CC1(CNC(C2CC(=O)N(c3ccccc3Cl)C2)=O)CCN(C(=O)CC2CC2)C1 N1(C(C(OCC)OCC)=O)CC2(C1)CN(C(=O)Cc1cccc[n+]1[O-])C2 CC1CN(C(=O)CCC2CC2C)CC1NC(=O)CCCn1ccccc1=O N1(C(C#C)C)CCN(C(=O)C(C)CNC(c2ncn(CC)n2)=O)CC1 C1(N(C(=O)Cc2cc(C)ns2)CCC)CCN(C(c2ccn(C)c2C)=O)CC1 c1(C(N2CCC(C(C)NC(C3C4COCC34)=O)C2)=O)ccc(O)cc1F N1(C(c2scc(C(C)=O)c2)=O)CC(CNC(c2ncccc2C2CC2)=O)CC1C Cn1nccc1NC(c1cnn(CC(F)(F)F)c1)=O c1(C(N2C(CN(C(c3cnnn3C)=O)CC)CCC2)=O)cnn2c1NCC(C)C2 c1(OC)cc2cc(OC)ccc2c2c1N(C(C1CC=CCC1C)=O)CCCC2 c1(C(=O)NCC2CCN(C(c3c(OC)nsc3OC)=O)CC2)cccn(O)c1=O N1(C(c2c(C)oc(C(C)C)c2)=O)CCC(C2CCN(C(c3ccccn3)=O)C2)C1 C1(NC(c2c(C)nc[nH]2)=O)CC(CNC(=O)Cc2cccn2C)C12CCC2 CS(=O)(=O)c1ccsc1C(c1nnnn1C1CCCC1)NCc1ccc(Br)cn1 N1(C(=O)CCN(C(c2ccncc2F)=O)C2CC2)CC2CCC1CC2 Cc1cc(NC(=O)C(N2CC3CC3(c3cccc(Br)c3)C2)=O)cc(Cl)n1 c1(NC(C2CN(C(c3cc(F)c(F)cc3Br)=O)CCO2)=O)cc(Br)c(O)cc1Br Cc1ccc2c(c1)CCC(C(=O)NC1CC(CO)N(C(=O)CC3OCCO3)C1)O2 C1(C(C)C)N(C(=O)CC2CCCC2O)CC12CCN(C(=O)C=CBr)CC2 CCC(C(=O)N(CC(C)(C)CNC(=O)CC(C)(O)COC)C)C(F)(F)F c1(C(CC(=O)NCC(CC)NC(C(C)=C(CC)C)=O)C)ccc(F)cc1 C1(CNC(=O)Cn2cccnc2=O)CN(C(=O)C2=CCS(=O)(=O)C2)C2(CCC2)C1 c1(C(N2CC(C)(NC(CC(CC)SC)=O)C2)=O)cc2cc(OC)ccc2[nH]1 c1(C(N2CCOCC(CNC(COCC(=C)C)=O)C2)=O)cccc(OC)c1C C(C1CCC(C)CC1)=C(C(=O)NC1C(SC)CN(C(C2(C)CCC(=O)C2)=O)C1)C CC(C)C(F)C(=O)NC1(NCCNC(=O)C(C)NC(C)(C)C)CCCCC1 C1(N(C(=O)Cc2cccnc2)CC)CCN(C(=O)Cc2nocc2C)CC1 c1(N(CC(C)O)CCNC(C2(C(=O)NCC)CC2)=O)cc(O)nc(O)n1 N1(C(=O)OC)CCN(C(C2C3COCC23)=O)CC(CO)C1 CC1(NC(C23CCC2CN(C(c2ccoc2)=O)C3)=O)CCS(=O)(=O)C1 c1(C(N(CCC)CCNC(c2csc(C)n2)=O)=O)cccc(-n2nccn2)c1 C1(CNC(C2(O)CC(C)(C)C2)=O)CC12CCN(C(c1cccnn1)=O)CC2 C(=O)(CCC(=O)C(C)(C)C)N(CC(C)C(=O)N(CC(=O)NC1CC1)C)C N(C1c2ccccc2CCC1F)C1(c2n(CCC)nnn2)CC2(C1)OCCO2 c1(C(C)C)ncc(CN(C)C(C2CCN(Cc3cccn3C)C2)=O)s1 C1(O)(CNC(C2(C(C)NC(=O)CC3CSCCO3)CCC2)=O)CCC(C)(C)C1 N1(C(C(C)NC(C)=O)=O)CCCC2(CC(NC(=O)Cc3cc[nH]n3)C2)C1 CC(=O)CCN=C(NCCC1CCCCO1)N1CCC(CC(F)(F)F)C1 CCCC(C)(C)CC(=O)NC1(C(=O)NCCC(C)C(C)(C)C)CC1C Cc1cnc(C(=O)NCC(F)CNC(=O)C(N2CCN(C)CC2)C)cc1C#N c1(C(=O)NC(CCCNC(CCC(=O)NCCC)=O)C)ccc2c(c1)CC(C)O2 c1(C(N2C(CN(C(CN(C)CCO)=O)C3CC3)CCC2)=O)cc(F)cc(N)c1F C1(NC(c2ccc(CC)o2)=O)CCCC1(C)CNC(=O)CC(C)SC N1(CCNCC(C)(C)CC2CC2)Cc2ccccc2C1 Cc1cc(C(N2CC(CNC(C3(C)CC3F)=O)C2)=O)cc(C)c1Cl N1(CCCNC(=O)C(=O)NCC2CC23CCOC3)C(=O)NC2(CCC2)C1=O c1(CC(=O)NC(CCCNC(CCC(=C)Cl)=O)C)ccc(CC)cc1[N+](=O)[O-] CCC(CCC(=O)NCCNC(=O)NC1CC1)NC(C1(OC)CCSC1)=O CC(C)CC(CC(=O)NCC(C)(C)C1CC1)NC(C1CC(=C2CC2)C1)=O N1(C(C)C(=O)O)CCC(c2ccccc2)C1 C1(CC(=O)NCC(CCNC(C2N(S(C)(=O)=O)CCC2)=O)O)CCCCCC1 c1(C(NOCc2cn(C(c3ccc(O)cc3)CC)nn2)=O)nc[nH]c2ncnc1-2 C1(F)(C(=O)OCC(CCOC)(C)C)CC2CCC1CC2 C#CC1(CNC(=O)C(CCCC)NC(=O)Cc2cc(C)on2)CCOCC1 C(=O)(CCCCC(N)=O)N1CC(C(C)NC(c2ccc(C3CC3)cc2Cl)=O)C1 C(=O)(C#CC(C)(C)CNC(=O)C(CC)CC)NC(C#C)(C)C c1(C(N2CC(CCNC(c3cc(CF)on3)=O)C2)=O)nncn1-c1ccccc1 C1(N(C(=O)CCC2(C)CC2)C)CCN(C(c2cc(C(F)F)nn2C)=O)CC12CC2 N1(C(c2cncc(OC3CCC3)c2)=O)CCN(C(=O)C2=CCSC2)C(CO)C1 c1(C(N2C(CNC(C(CC)N(C)C)=O)C=CC2)=O)ncc(OC)nc1OC N1(C(CC2CN(C(C)=O)C2)=O)CC2CC(NC(C(C)C(=O)N(C)C)=O)CC2C1 C=C=CC(C)C(=O)NCC1(O)CCN(C(C2(CO)CC(F)(F)C2)=O)C1 Cc1ccc(CNCC(c2ccc(F)c(F)c2)N)nc1C CCCC(O)CC(=O)NC1CCCC1CNC(C1CC(C)CC(C)C1)=O C1(CNC(Cc2ccc(C)cc2)=O)CN(C(C2(F)CC=CCC2)=O)CC12CC2 C(=O)(CCC(=O)N(C1(SC)CN(C(=O)C(C)(O)C2CCC2)C1)CC)NCC CC1CN(C(c2cn(-c3cccc(OC4CCOCC4)c3)nn2)=O)CCN(C)C1 C1(C)(CCC(=O)N(C(CCSC)C)C)CN(C(c2csnn2)=O)C1 c1(C(N2CC(CC)C(NC(=O)C(=O)N(C)C)C2)=O)cccc(C)c1-n1cccc1 C1(NC(C2(C)CCOCC2)=O)COC2CN(C(c3cn(C(C)(C)C)cn3)=O)CC12 Cc1nc(C)n(O)c1C(=O)NCC1CCCCN1C(=O)Cn1cc(C2CC2)cn1 N1(C(c2c(C)nc(C(F)(F)F)s2)=O)CCN(C(C2CC3CCC2O3)=O)CC1C c1(C(N2CCC(NC(c3c(CC)onc3)=O)(COC)C2)=O)ccc(C)c(C)c1 C=CCC(CC=C)C(=O)N(C)CC1CCCN(C(=O)CCCCCCC)C1 C1(C)(N(CC(N)=O)C(C)=O)CCN(C(C2CNC2)=O)CC1.c12cccc(c1)SC2 C1(C(=O)NCC2(CNC(C3CCC4(CC4)C3)=O)CC2)CCC2C(C1)C2(F)F N1(C(C(C2(O)CCCCC2)NC(C2CSCC(=O)N2)=O)=O)CCC(O)C(F)(F)C1 N1(C(Cc2cncc(C)c2)=O)CC(C(=O)NCC(C)(C)C)C(C)(C)C1 CCCC(O)C(CO)NC(=O)NCc1ccc(O)cc1C CC(C)CC(C)(C)NC(C1CCCN1C(=O)CC1CC2C=CC1C2)=O C(=O)(C(Cc1cc[nH]n1)NC(=O)C(C)C1(OC)CCC1)N(C(C(C)SC)C)C CC(C)(C)CCC(=O)N1CCCCCC1CNC(=O)CC(C)(C)c1cccs1 c1(CC(=O)NCCN(C(=O)C(F)CC2CCC2)CC)cnc(C(F)(F)F)s1 CCC(CC)CCCC(=O)NCC1(O)CC(CNC(c2cnn[nH]2)=O)C1 C(=O)(C1=NOC2(CCOC2)C1)NCCCC(C)NC(c1c(F)cncc1Cl)=O N1(C(CC(C(=C)C)OCC)=O)CCCC2(NC(=O)COC3CC(F)(F)C3)CC2C1 C1(NC(C(COC(C)C)NC(C)=O)=O)C2CCC1N(C(c1cnnn1C)=O)C2 Cc1nc(N2CCCN(C)CC2)ccc1NC(N1CC(CO)CC1C)=O Cc1ccc(CCC(=O)NC(CCNC(C2OCC2(C)C)=O)C(C)C)cc1C C(=O)(C(F)C(C)(C)O)NCCCOCCCNC(C(COC)(C)OC)=O C(CCCCCCNC(C1(C)CC2CCC1C2)=O)n1cc(CN(C(C)C)C)nn1 C(=O)(C1=NNC(=O)C1)NC(CCSC)C(=O)NC1CC12CC(O)C2 N1(C(C2CCC(=O)N2)=O)CCC2(CCCN(C(=O)C=CC3CCOCC3)C2)C1 c1(C(=O)NCCCCCN(C(c2nccc(C)n2)=O)C)cc2ccccn2c1 c1(NCC2CCN(C(C=Cc3ncn(C)c3)=O)C2)nnc2c(c1C#N)CCCC2 c1(C(N2C(C(=O)Nc3c(F)ccc(C)c3)COCC2)=O)ccc(O)c(F)c1 c1(C(=O)NCC2C(C)CCN2c2nncs2)cc(O)nc(Cl)c1 N(C1CCCc2cccnc21)(CC(C)C)C(=O)NC1CCCC1(C)O CC1(C)CC(CNC(=O)C=CC2CCCN2C(c2ccc(O)cn2)=O)CO1 c1(C(=O)NCC(C)(O)CNC(=O)Cc2ccco2)c[nH]c2ccncc12 N1(C(c2c(C)nc(C(F)(F)F)s2)=O)CCC(C)(NC(C2CC(C)(C)CO2)=O)CC1 C1(CNC(C2(C)C(C)OCC2)=O)CN(C(=O)Cc2ccc(Cl)s2)CC1(F)CO N1(C(C2C(CC)C2)=O)CCC(CNC(=O)COCC(=O)NC)(OC)CC1 C(=O)(C(C)S(N)(=O)=O)NCC1C(NC(C2CCN(CCC#C)CC2)=O)CC1 N1(C(CC(C)N(C(=O)CCCC#N)C)=O)CCC2(CCOC2=O)C1 C1(CC)C(C(=O)NCC2CCCCC2)CCCN1C(C1CCCCC1O)=O CC(C(CO)NC(c1cnn(C2CC2(F)F)c1)=O)NC(=O)COc1ccccc1 C(CC(F)(F)Cn1cc(C2(O)CCOCC2)nn1)NC(CC(C)NC(N)=O)=O C1(C(N(CCNC(=O)CC(=O)NCCO)CC)=O)CN(C(=O)C2CC2)C2CC12 N1(C(CCCn2c(C)ncc2)=O)CCCC(C2CN(C(C3(Br)CC3)=O)C2)C1 C1(C(N(C(C(CC)C)C)C2CC2)=O)CCN(C(=O)c2ccc(N)cn2)O1 C1(CC#C)(C(=O)NC)CCOCC1.C(=O)(C(C#N)CC)NCC1(N)CCC1 c1(Cc2cn(C3C(C)CN(C(=O)C4=CCCCO4)C3)nn2)c[nH]nc1S(N)(=O)=O c1(C(N2C(CNC(C(CCOC)C)=O)COCC2)=O)nnn2c1CCC2 C(C1CN(C(C2CC2(Cl)Cl)=O)CC1C(=O)NCCCc1ncco1)=CC C1(C(C)(C)NC(c2cocn2)=O)CCN(C(=O)Cc2cccc(F)c2)CC1 c1(C(=O)NC2CC(CNC(=O)Cc3nc[nH]n3)CC2O)cc(C2CC2)ccc1F N1(C(C2CC(C)OC(C)C2)=O)CC2(CCCC2NC(c2ncccc2N)=O)C1 C1(Cl)(C(=O)NCCC(C)N(C)C(C2CC(C(F)F)C2)=O)CC1(F)F C(C(=O)N1CCC(C(=O)NCC2(C(N)=O)CC2)(COC)C1)(C(C)C)OCC N1(C(CCC=CC)=O)CCN(CCN(C)C(c2cn(C)nc2Br)=O)CC1 C(C(F)(F)C(F)(F)F)OCCC(=O)N(C(CNC(C1C(=C)C1)=O)C1CC1)C C1(C(=O)NCCCn2c(C)ncc2)CCCCN1C(=O)CCc1csnn1 C1(C(N2CC3(CCC(CNC(C(C)C)=O)O3)C2)=O)COc2ccccc2O1 C1(C(N2CC(OCCN(C(=O)Cc3ccsn3)C)C2)=O)CC2C=CC1C2 N1(C(c2ccc(SCC)cc2)=O)CCCCC(CNC(=O)CN(C)CCO)C1 c1(C(N2CCC(N(C(CNC=O)=O)CCO)C2)=O)nccc2c(Cl)cccc12 C1(NC(=O)NCC(C)OC)CCN(c2ccc(C(F)(F)F)cn2)CC1 c1(C(=O)NC2C(NC(=O)C3=CSCS3)COCC2)ccc2cnccc2n1 C(=O)(CCCC(C)C)N(CC(C)(CO)N(C)C)SC.c12coc(n1)CC(=O)C(=O)C2 c1(C(=O)NC2C(NC(C(C(CC)O)C)=O)C2)cc(S(C)(=O)=O)cc(C)c1C C(=O)(CCCN(C(=O)C=C1CCC1)C)NC(CN(C)C)(C)C c1(C(=O)NC2CCCC2NC(c2n[nH]cc2F)=O)ccc2c(c1)CCC(O)C2 N1(C(c2c(CC)cc[nH]2)=O)CCC(C(N2CCC(C(CC)CC)C2)=O)C(O)C1 N1(C(C(CC)O)=O)CCC(C)(CNC(c2ccc(COC)c(F)c2)=O)CC1 C1(NC(c2c(C)cc(CC)o2)=O)CCC(C)N(C(=O)Cc2ccc(C)cc2C)C1 c1(NC(C2CCCN(Cc3ccc(C(=O)OCC)o3)C2)=O)c(Br)cc(Br)c(O)c1Br c1(N(CCOCCNC(C(C)OC2CCOC2)=O)C)nccn1C.C1CS1 N1(C(c2cn(C)nc2)C(=O)NCCOCC2CC2)CC2C(C1)C2(F)F c1(SC)nccc(C(=O)NCCOC2CCN(C(=O)C=Cc3ccn(C)c3)C2)n1 Cc1nn(C2CCC2)cc1C(=O)NCCC1CCCN(C(C2(CCO)CC2)=O)C1 C1(NC(c2cn(CC)nc2C(C)C)=O)CCC(C)N(CC(O)COCCOC)C1 C(=O)(CCC(C)(C)C)N1C(CN(C(=O)CC(c2c(C)n[nH]c2C)C)CC)CCC1 C(=O)(CC(C)C(F)(F)F)NC(C1CN(C(c2c(C)nc[nH]2)=O)C1)C CCCCCC(F)C(=O)NC1C=CC(C(=O)NC2CCC(CCC)CC2)C1 c1(C(N(C)CCNC(=O)C(O)Cc2ccccc2Br)=O)ccc(F)c(F)c1 CN1CCCCC1CC(N1CCOC(C(N)=O)C1)=O C1(NC(C(COC)O)=O)CC12CCC(NC(C1(O)CCSCC1)=O)CC2 N1(C(c2n(CC=C)ccc2)=O)CC2(CC(NC(=O)CCC(=C)Cl)C2)C1 c1(C(=O)NC2(CC(N)=O)CCN(C(C(CC)SC)=O)CC2)cc(F)c(N)c(F)c1 C1(C(=O)NC2CCC23CN(C(=O)COCCc2cccs2)C3)CCC2(CCC2)O1 C#Cc1ccc(C(=O)NC(c2cccnc2)C(=O)NCc2ocnc2C)o1 c1(CNC(C(CN(C)C)NC(C(C)OCCC(C)C)=O)=O)ccc2c(c1)CCC2 N1(C(c2nc(C)oc2)=O)CCCC12CCN(C(=O)CCC(C)N(C)C)C2 Cc1cc(C(=O)NCC2CN(C(=O)CCF)CC2C(F)(F)F)c(O)nn1 c1(-c2cn(C(C)C(N3CCNC(=O)C3CCO)=O)nn2)c(F)ccc(F)c1Cl n1(C(C)C)cnc2c(NCCc3ncccc3F)[nH]c(=NCC3CC3Cl)nc12 N1(CC(=O)NC(C2CC2C(F)(F)CC)=O)CCC(CCCC2CC(CC)C2)C1 C=C1CCN(C(=O)C(C)OCC2CC2)C(C(=O)N(CC(=O)OC)CCC)C1 C1(NC(CC2CCCC(C)(C)O2)=O)CCNCC2(CC2)C1 C1(CCC)CCC(C(=O)NC23CC(CNC(C4(C#N)CC4(C)C)=O)(C2)C3)CC1 c1(C(N2CC(N(C(CCC=C=C)=O)C)C(C)(C)C2)=O)coc2ccccc12 n1(Cc2nc(CCCCCC)nn2-c2ncnn2C)nc2c(n1)CCCC2 CC1(C(=O)Nc2cnccc2I)CCN(Cc2ccc(Br)c(Cl)c2)CC1 C(=O)(C(C)(C)C(O)C(C)C)NC1CC(N(C(c2c(C)c(Cl)cnc2)=O)C)C1 c1(CNC(C(c2cccs2)N(CCC)CC)=O)ccccc1Br C1(C(N2CC(C)N(C(=O)CC#N)CC2)=O)CCc2cnn(C)c2C1 C(C)(C)(C(C)CC(=O)N(CCCO)CCO)NC(c1cccc(CC)c1)=O C(=O)(C1=C(F)CN(C(=O)CC(C)C(F)(F)F)CC1)N(C(C)C)CCF C#CCC(CC(=O)OC)NC(C1CNC(=O)CN1C(=O)C1=CCCSC1)=O CC1=Nc2ccc(C(=O)NC3CC(O)C3)cc2C1(C)C C1(NC(=O)OC(C)(C)C)CCCN(C(=O)NC(CC2CCCC2)CO)C1 C(CO)(CCCNC(C1CC2C=CC1C2)=O)NC(c1ccc(C2CC2)cc1)=O C#CCC(C)(C(=O)NCC(C)(C)COC)NC(=O)CNC(=O)CC N1(C(=O)OC(C)(C)C)CCc2cc(C(N3CC(c4ccncc4O)C3)=O)ccc21 N1(C(CN(CC)CC)=O)CCC(CC(C)NC(c2cnsc2)=O)CC1 c1(C2C(C)C2)ccc(-c2nc(C3(C)CCCO3)no2)cc1 CCCC(C)(O)C(=O)NCCC1CN(C(C2CC3CCC(C2)O3)=O)CC1C C1(C(=O)NCCCc2cc(C)no2)C2CCC(C2)N1C(c1cc(=O)cc[nH]1)=O N1(C(c2cc(=NC)[nH]cc2)=O)CCC2CCN(C(=O)CSC(F)F)C2C1 C(=O)(C1=CC(O)C(NC(C2CN3CCN2CC3)=O)C1)N1CC(CC(C)C)OCC1 c1(N2CCN(C)CCN(C)CC2)nc(=NC2CCC(O)C2)[nH]c2ccccc12 C1(NC(C2C(NC(C(C)c3cc[nH]n3)=O)CC2)=O)CCCC1(F)F C#CCCCCC(=O)NC(C)CCN(C)C(c1cocn1)=O c1(C(=O)NC2(CNC(C(C)(C)C3CCCO3)=O)CC2)ncccc1F c1(O)cc(F)ccc1F.N12CC3C(C3C1)NC2=O.C1(C(=O)OC)CCN(C(=O)N)C1 CCC(F)(F)C(C)(C)C(=O)NC1CN(C(=O)COCC2CCCO2)CCC1CO C1(C(=O)NCC23CC(NC(COCCC)=O)(C2)C3)CC2(C1)CS(=O)(=O)C2 C1(C(=O)NC(CCOC)C)CN(C(c2cncc(OC)c2)=O)CCO1 Cc1cc(F)c(C(=O)NCCCN(C(c2ccc(S(C)=O)cc2)=O)CC)cc1F c12cc(ccc1[N+](=O)[O-])NCCCN(c1nc(C)cs1)C(=O)C(C)O2.CCOC c1(C(=O)NCCC(=C)CNC(=O)C(c2cccc(Cl)c2)SC)c[nH]ccc1=O C1(NC(C2(COC)CN(C(=O)CC3COCC(C)O3)C2)=O)CCCCCC1O CC1COCC(C(=O)NC(C(N2CC3C(CO)C3C2)=O)C2(O)CCC2)O1 CC1C(C(=O)NC2COC(C(F)F)C2)CCN1C(=O)C1=CCCC1 c1(CC(C)C(=O)NC2CCC(NC(=O)CCC(C)N(C)C)CC2)ccc(Cl)cc1 C1(NC(C(C)S(C)(=O)=O)=O)CCCCC12CCCN(C(=O)CN1CCCC1)C2 N1(C(c2[nH]c(=NCc3cnc(C)nc3)sc2)=O)CCC2(CC1)CNC(=O)C2 c1(C(=O)NCC2(C)CCN(C(=O)C(O)CF)C2)ccnc2ccnn12 C1(N(CCC#N)C)C(=O)NC1Cc1ccccc1.C1(C(=O)OC)(COC)CC1 C=CC(C)(O)CC(=O)N1CCN(S(C)(=O)=O)C(CC(F)F)C1 N1(C(c2nc(C(C3CCCO3)C)sc2)C(=O)NC)CC2CC1(C(=O)OC(C)(C)C)C2 CC(C)C(O)CC(=O)NCCOCCNC(C1CCCN1C(c1ccsc1)=O)=O C(=O)(CCC(C)(C)C)NCC1(CNC(c2ccc(CCCC)cc2)=O)CCC1 C1(C(=O)NC(CC)CNC(c2cccc(C(C)=O)c2)=O)CN(C)CCN(C)C1 C1(NC(C(C2(C)CC2)NC(C2(CC3CC3)CCCC2)=O)=O)CC12CCCCC2 N1(C(c2cnc(CC)s2)=O)C2CCC1CC(N(C)C(c1cccc(F)c1F)=O)C2 C1(C(N2C(CNC(C(C)C(C)c3ccc(Cl)cc3)=O)CC2)=O)COCCN1C=O c1(C(=O)NC2CCC(C(=O)NCC)C2)nc(OC)c(C)s1 c1(N2CCC(c3cc(C)[nH]n3)C2)nc(=NCC(C)c2ccsc2)[nH]c2ccccc12 C1(C(N(CC(C(=O)N(CC(C)N(C(C)=O)C)C)C)C)=O)CCC2(CC2)C1 Cc1cccnc1C(F)(F)C(=O)N(C)CC1CCCN(C(C2OCC2(C)C)=O)C1 N1(C(c2cn(CCOC)nn2)=O)CC2(CCC(CNC(c3cocc3C)=O)O2)C1 Cc1cccnc1C(=O)N(C1CN(C(c2ccccc2-c2cccnc2)=O)C1)C CC(C1CCCCC1)=CC(=O)NC(C)(CNC(c1nnc(C)s1)=O)C1CC1 c1(OC)ccc(C2CCCN(C(=O)NC3(c4ccc(=O)n(C)c4)CC3)C2)cc1OC N1(C(Cn2c(CCC)ncc2)=O)CCC(C)C(NC(c2sncc2C)=O)C1 C(C(=O)NCCc1ccc(CNC(=O)C(c2cncnc2)C)cc1)(C(C)C)OC Cc1c(C(=O)NCCN(C)C(c2occc2F)=O)nn2c1CCCC2 C1(N(C(C(c2ccc(F)cc2)OC)=O)C)CCCN(Cc2cnc(=N)[nH]c2)C1 C1(O)(CNC(CCC=C)=O)CCN(C(C2OCCCC2c2ccccc2)=O)CC1 N1(C(c2cccc(F)c2O)=O)CC2(CCCN2C(=O)CC(F)(F)F)C1 N1(CCCCOC(C(CC)O)=O)CCCC(CN(C)C)C1 N1(C(C(CC2CC2)OC)=O)C2CC1CN(C(c1cc(O)cc(F)c1)=O)C2 N1(C(CC(CC)SC)=O)CCN(c2ccc(OC)cc2)C(=O)C1 CC1C2CC(C2NC(=O)CNC(c2ccoc2)=O)N1C(c1cc(Br)c[nH]1)=O Cc1cc(C(N2CCN(C(=O)C(C)CCO)CC2CCO)=O)nnc1C CC(O)CCCc1cn(CC2CCNC2)nn1 CCCCC(CNC(C1(C)CC=CCC1)=O)NC(C1CC(N(C)C)C1)=O Cc1nc2c(o1)CCCC2CC(=O)N1CC(NC(=O)C2=COCCO2)CC(F)C1 c1(C(=O)NC2CN(C(C3CCN(CC)CC3)=O)C3C2C3)ccc(SC)cc1C c1(NCCNC(N2C(c3nc(C)sc3)CCC2)=O)cccc(I)c1 Nc1cc(F)cc(Cl)c1C(N1CCN(C(c2ccccn2)=O)C(C2CC2)C1)=O Cc1ccc(C(=O)C(=O)NC2CCC(CNC(c3[nH]nnc3C3CC3)=O)C2)cc1 c1(C(N(CC(C)NC(C(CC)(C)C(N)=O)=O)C)=O)cc(=O)c2ccccc2[nH]1 C(=O)(C(C(C)(C)C)n1ccnn1)N1CC(NC(c2cc(N(C)C)ncc2)=O)C1 N1(C(CCC#C)=O)CC2CC(NC(c3cccnc3SC(F)(F)F)=O)C(C2)C1 C1(CC(=O)NC2CC(NC(CCc3c[nH]c(=N)[nH]3)=O)C2)CCN(CCF)CC1 N1(C(=O)Cc2cnsc2)CCC2(C1)CN(C(C1CC13CCCOC3)=O)C2 c1(C(N2CC(N(C(CN3CCCC(CC)C3)=O)C)C2)=O)ccc(F)cc1C(F)F C12(C(=O)NC(C3CCCCN3C)C)CC(CO)(CN1C(=O)CCCc1cnn[nH]1)C2 C1(CNC(C(CC)F)=O)CN(C(C2(COC)CC(F)(F)C2)=O)CCCO1 CC(O)CC(C(=O)O)NC(=O)CC1CCCCC1C N1(CC(=O)NC2C(CNC(CC=CC=C)=O)C2)CCCC1CO C1(OC)CN(C(=O)CSC2CCCC2)CC1CNC(=O)COCc1csc(Cl)n1 c1(N(C(CCC#C)Cc2ccccc2)C(C)=O)ccc2c(c1)CCC2 N1(C(CC2CNC(=O)O2)=O)CCCC12CCCN(C(=O)COC(F)F)C2 C(C(C)C)(C(O)C(=O)N1CCN(C(c2ccc(=N)[nH]c2)=O)C(CO)C1)OC N1(C(c2c(C)[nH]cc2)=O)CC2CC1CCN2C(=O)C(C)CC1CCCCC1 c1(C(N2CCC3(C(C(N4C(C)COCC4)=O)C3)C2)=O)cc(Cl)c(Cl)c(Cl)c1 C1(C(C)C)CCC(C(=O)NCC2(C)CNC(=O)O2)N1C(c1ncc(F)cn1)=O C1(NC(=O)CC2(CO)CC2)CN(C(=O)C(=C2CCCCC2)F)C2(CCC2)C1 C(=O)(C(C)CCC(C)(C)C)NC1CC(C)N(C(=O)C(C)(C)F)C1 c1(CNC(C2N(C(C(C)Cn3ccnc3)=O)CC2)=O)c(Cl)cccc1Cl CC1CN(C(=O)COc2cccc(Cl)c2)CC1CNC(=O)CCn1cccn1 c1(N2CC3C(NC(CC(C)(O)C(F)(F)F)=O)C3C2)cc(Cl)nc(S(C)(=O)=O)n1 N1(C(C(C)N(C(C)=O)C)=O)C2CCC1CC(O)(CNC(C1CC(O)CN1C)=O)C2 C(C(C)(C)CNC(c1cnns1)=O)N(C)C(c1ccc(C(F)(F)F)o1)=O C(CCCC(=O)NC1(CN(C)C)CC1)N(C(CNC(C1C(C)C1)=O)=O)C N1(C(c2cc[nH]c2C2CC2)=O)CCN(C(C2(F)CCOC2)=O)CC1CO C1(C(=O)OC)CC2(CCCN2C(=O)C(N)CC2CCS(=O)(=O)C2)C1 CN1C(=O)Cc2ccc(C(=O)NCC3CCCCN3C(=O)Cn3cnnn3)cc21 Cc1cn2cc(C(N3CC4(CCCC4NC(c4cnn(C)c4F)=O)C3)=O)nc2s1 N1(CCc2c(C)n[nH]c2C)CCCC(C)(C(=O)NCc2ncc(Cl)s2)C1 C(CNC(=O)CN1CC(C)(C)C1)(C(C)C(C)C)Nc1ncc(C(=O)OC)cn1 c1(CCC(=O)NCC2CCN(C(C3OCCCO3)=O)C2)cccc2c1OCCO2 N1(C(c2ccc(C(C)=O)cn2)=O)CC(NC(=O)CC2CCC(C)C2)CC2(CC2)C1 Cc1cc(C(=O)NC2CC(O)CN(C(c3cncc(F)c3C)=O)C2)c(O)c(C)c1 CC1CC(C(=O)NCc2cccc(C(=O)NCC[Si](C)(C)C)n2)CCO1 c1(CCC)cc(C(=O)N(C)CCN(C(=O)CCC2CC(C)(C)CO2)C)ccn1 N1(C(c2scc(C)c2Cl)=O)CCC(NC(C2CCC(=O)N(C)C2)=O)CC(O)C1 Cc1cc(C(=O)NCCCC2CCCN2C(c2cc(Cl)n[nH]2)=O)c(O)nn1 C(=O)(C1=CCCN(C(=O)CC2CCC(=O)N2)C1)N1CCCC(C(=O)NC)C1 N1(C(c2c(SC)nccn2)=O)CC2CCCC(NC(C3CCCSS3)=O)C2C1 c1(C(=O)NCC(CCNC(C(C(C)OC)N(C)C)=O)O)cccc2[nH]ccc12 C#CCC(O)C(=O)N1CC=CC1(C(=O)N(C(C)C(=O)OCC)C)COC CCCC(C(=O)NC1(CC)CC(C)(C)C1)NC(C1CCN(C(C)=O)C1)=O Cc1ccc(S(C)(=O)=O)cc1C(=O)NC1CCN(C(c2nc(Br)c[nH]2)=O)C1 Cc1cccn2nc(C(N3CCC(NC(c4ccc(F)c(Cl)c4N)=O)C3)=O)cc12 C1(C(=O)NCC(CC)NC(c2cccc(N(C)C)c2)=O)CCC2(CCC2)OC1 c1(C(C)=O)c(C(=O)NC(C)CCC(=O)Nc2ccc(C(C)C)cc2)cnn1C C1(OC)CC(CNC(c2nccn2C)=O)N(C(=O)CCCn2cccc2)C1 Cc1cnc(CNC(=O)C(F)CC2CN(C(=O)CCC3CCC(=O)C3)C2)o1 C(=O)(C(C#N)C(C)C)N(CC(C)N(C(c1nccc(CC)c1)=O)C)C C1(C(=O)NC(CNC(c2c(C)nns2)=O)C2CCC2)NC(=O)C2CCC12 c1(C(N2CC3C(C(=O)NC(CC)(C)C)C3C2)=O)cncc2cnccc12 C(=O)(C#CC1(C)CCCO1)N(CC)CC1CCCN1C(=O)CC1CCCN(C)C1 c1(C(N(CCC(=O)NCc2cc(C(C)C)no2)C2CC2)=O)cn(C)c(=O)n1C N1(C(CC(=C=C)C)=O)CCC(C2(NC(C3CCc4nnc(C)n4C3)=O)CC2)CC1 c1(CC)ccc(C(=O)NCC2CCN(C(c3ccc(C)cc3F)=O)CC2)c(C)n1 c1(C(=O)NCC23CC(NC(CC(C)N(C)C)=O)(C2)C3)c(Cl)ccc2c[nH]nc12 c1(CNC(C(C)n2ccnn2)=O)cc(C(=O)N(CC(C)O)C2CC2)on1 N1(C(C(C)C2(O)CCC2)=O)CCC(O)(CCNC(=O)CCOCC(F)F)C1 S(=O)(=O)(c1cnc(Cl)c(Cl)c1)N(c1ccc(F)cc1)CC c1(N(CCC(N2CC(CNC(CN(C)C3CC3)=O)C2)=O)C)nc2ccccc2s1 N1(C(CCSCC)=O)CCC2CC2(C(=O)NCc2nn(C)cc2CO)CC1 C#CCN(OC)C(=O)C1C=CC(NC(C2CC2CC(C)C)=O)C1 CCN=C(NCc1nnc(CC)s1)NCC1CC1(F)F C12CCC(CC1)CNC2=O.C1(CN(C)C(C2CC(C)(C)CO2)=O)CCCC2CC12 CC(C)CC(CNC(C1CC(F)C(=O)N1)=O)NC(C1CCC(n2cccc2)CC1)=O N1(C(c2cnn(CCC)c2C)=O)CC(NC(=O)CP(C)(C)=O)C2(CC2)C1 c1(C(=O)NC(C(=O)NC2CC(C)(C)OCC2)C2(O)CCC2)c[nH]c2nccc-2c1 CC1(C)CCOC(CC(N2CC3(C(=O)NCC4CC(O)C(O)C4)CC2CO3)=O)C1 N1(C(Cc2ncc(C)s2)=O)CCOC2(C1)CN(C(C1(C)CC3(CCC3)C1)=O)C2 N1(CC(CC)OC)CCCC(NC(c2n[nH]c(C)c2C(F)(F)F)=O)C1C CC(C)C(C)(CNC(C1CCS1(=O)=O)=O)NC(c1ccccc1CN(C)C)=O N1(CC(=O)NC(C2CCCN(C(c3nn[nH]c3Cl)=O)C2)C)CC(=O)N(C)C1=O c1(C(=O)NCCC2N(C(CC(=O)OCC)=O)CCC2)ccc(C#CC2CC2)cc1 c1(C(C)C)c(N(C)CC2CCCN(C(=O)C(C)OCC3CC3)C2)ncnc1Cl C=C1CCC(C(N2C(C(=O)NC(C)(C)CO)CC3CC23)=O)CC1 C1(C(=O)NC2C(C)N(C(c3cccc(F)c3)=O)CC2)CCC2CCCCN12 CCC(CCC(=O)NOC(C)CC)NC(=O)C(C)(C)c1ccno1 C1(CNC(=O)CC2CCCCO2)CCN(C(c2cn(CCF)nn2)=O)CC1(F)F c1(C(N(CC(CNC(C(c2ccc(F)cc2)C)=O)(C)C)C)=O)ccc(N)cn1 N1(CCC(=O)NC2C(NC(C3(Br)C(C)(C)C3)=O)CCC2)CCCCC1=O C(C(C)(C(C)C)NC(=O)CC1(C(=O)Sc2nc(C)[nH]n2)CC1)NC(CN(C)C)=O C(CS(=O)(=O)CC(=O)N1CC(C2CN(C(=O)Cc3cnn(C)c3)CCO2)C1)OC C1(CNC(=O)CCc2nccs2)(CNC(=O)CC2(CO)CC2)CC12CCC2 C(C(C)(C)CC(=O)NCC(CC(C)C)NC(=O)CC1(C)CC1(Cl)Cl)OC CC1OCCN(C(C2CCC3CC23)=O)C1C(=O)NC1(C)CCCCC1 Cc1ncn(C)c(=O)c1C(=O)NC1CN(C(c2csnc2Cl)=O)CC1C c1(CC)ccc(C(N2CC(NC(=O)CC3(CSC)CC3)C(C)C2)=O)c(C)n1 C1(NC(CC2CCCC(C)(C)C2)=O)CCN(C(c2ccc(C#N)o2)=O)CC1(C)C c1(C(=O)NCCC2(OC)CN(C(c3cc(C)cs3)=O)C2)cc(O)ccc1Cl c1(CC)ccc(C(=O)N(CC(C)O)CCNC(=O)CCN(C)CC)s1 N1(C(C2=C(C)CCC2)=O)CCC2(CCC(NC(C3CC(n4cccn4)C3)=O)C2)C1 c1(C(N2CC(CNC(CC(CN(C)C)O)=O)C(O)C2)=O)cccc([N+](=O)[O-])c1 c1(C(=O)NC(CNC(C(CCSC)O)=O)C(C)C)ccc(F)c(O)c1 c1(N(C(=O)CNC(=O)CNC(=O)C(O)CC2CCCC2)C)sccc1C#N n1(C(C)C)cnnc1CCNC(c1nc(C2CC2)cs1)=O C12(C(N3CCCC(C(=O)Nc4c(C)ccc(F)c4)C3)=O)CC3CC(CC(C3)C1)C2 Cc1nc(C(=O)NCC2(F)CN(C(c3ccnn3C3CC3(F)F)=O)C2)co1 C=CCC(F)(F)CN(C)C(C1CC(NC(=O)COCCCOC)CCO1)=O C1(CC(=O)NCC(CN(C(c2c(CC)non2)=O)C)C)CC2(CCC2)CO1 c1(OC)c(C(=O)NCCN2CCN(C(=O)Cc3ccns3)CC2)csc1C C1(C)(CNC(c2ccn(CCOC)n2)=O)CCN(C(=O)COC2CCCC2)C1 Cc1c(NCCc2cc(F)cc(F)c2)ncnc1NC1CCCC1CCC(C)C c1(CNc2n(C(C)(C)C)ncc2C(=O)O)c(Cl)ccnc1F c1(C(N2CCN(C(C3ON=C(C)C3)=O)C(CCO)C2)=O)ccc2cc(C)cn2c1 N1(C(C2(C)CCN(C(=O)CCc3ccccc3)CC2)=O)CC2C3CCC(C3)C12 Cc1cccc(C(=O)NC2(CO)CCCN(C(C3CC4(C3)CC(F)C4)=O)C2)c1C CC(C)(C(=O)NCCOC1CCN(C(C2C=CCC2)=O)C1)c1cccs1 C(CCC(C)C(=O)NCCCC1CCCN1C(=O)C(C)C(C)C)OC CC(C)C(C(C)NC(=O)Cn1nnc(=O)[nH]1)NC(=O)C=Cc1cn(C)nn1 c1(OCCC(=O)NC2C(CNC(CSC)=O)COC2)cccc(F)c1 N1(C(C(CC)COC)=O)CCC2CCN(C(C3CCC(O)CN3C)=O)C2C1 N1(C(CC2(CC)CCC2)=O)CC2CC(C)N(C(=O)C(C)c3ccco3)C2C1 n1(C2CC(NC(=O)Nc3ccnn3Cc3ccc(Br)cc3)C2)ncc([N+](=O)[O-])n1 C1(CNC(c2c(C)ncn2C)=O)CN(C(=O)CSC2CCOC2=O)CCC1C c1(OC)ccc(C(N2CCCC2C(C)NC(c2occc2C)=O)=O)cc1 C1(NCc2cn(C(C)C(N3CCCOC(CO)C3)=O)nn2)CCN(C)CC1(C)C C1(C(=O)NC(CCCC)CNC(c2nonc2N)=O)CS(=O)(=O)CC12CC2 CCC(CC(=O)NC(C)CC1CN(C(=O)Cc2cccc(C(F)(F)F)c2)C1)OC C1(C(=O)NCC2(C)CCN(C(C3CCCC3)=O)CC2)COc2ccc(Cl)cc2C1 C1(C)(c2cn(C(C(=O)N(CC(C)C)CCC#N)C)nn2)CCOCC1 N1(C(CCn2ccc(C)n2)=O)CC(NC(=O)C(c2ccc(Cl)cc2)CO)C(C)C1 C(CCCC(=O)N1CC(F)CC1CC(=O)N(C(C)CCO)C)OC C1(C(C)C)C(NC(=O)CCCNC(=O)C2CC2)CCN1C(c1ncn(C)n1)=O Cc1sc(C(=O)NC2COCC2CNC(=O)CCn2cnnn2)cc1[N+](=O)[O-] C=CC(C)(O)CCCC(C)C(=O)N(CC(C)(C)CNC(c1cccn1C)=O)CC C(C)(CCC(=O)NCC1(C)CC1)NC(C(n1ccc(C)n1)C)=O Cc1cccc(Cl)c1-n1nc(CO)nc1C1CC1c1cc(OC(F)F)cc(OC)c1 c1(C(=O)NC(C)Cn2cc(CN3CCCC3CO)nn2)cc2cc(Cl)ccc2o1 C#Cc1cncc(C(=O)NC2CC3CCC2(NC(=O)CC2(OC)CCCC2)C3)c1 O=C1CC(C(N2CC(C(N3CCC(C(F)(F)F)C3)=O)C2)=O)CN1 c1(C(N2CCC(NC(C(CC=CC)C)=O)C2)=O)c(N)cccc1Cl C1(C)(C(=O)NC(c2nccn2C)C)C=CCN1C(c1ccc(CO)o1)=O c1(NC(C2N(C(C(CC)OCC)=O)CC=C2)=O)ccc(O)cc1 Cc1nnn(CC(=O)NC2CC(CCNC(=O)C(C)(C)n3cnnn3)C2)n1 C(=O)(C(O)CC(C)C)NC1(C(=O)NC(CC)CC)CCSC1 C(=O)(C(C)C(F)(F)F)NC1C(OC)CN(C(=O)Cc2ccccc2Br)C1 C1(NC(C2CCC(Cc3cn(CC(=O)OCC)nn3)CC2)=O)CCC(C)(C)CO1 c1(C(=O)NCC2N(C(c3[nH]cc(-c4[nH]c(=N)sc4)c3)=O)CC2)ccccc1F c1(C(=O)NC(C(=O)NCC(CC(C)C)C)C2CCCO2)ccn(C)c(=O)c1 N1(C(C2(C(C)(F)F)CCC2)=O)CCC(O)(CNC(=O)C=Cc2ccc(Cl)s2)C1 C1(C(=O)NCC(C(C)C)(C)C)CC(O)C(O)CC1CNC(C1CCS(=O)CC1)=O C1(CC)(NC(c2cccc(C#N)c2)C)Cc2ccccc2C1 C1(NC(C2CN(C(CC(C)F)=O)C(C)(C)C2)=O)CCC(C2CC2)CC1 C#Cc1cnn(C)c1C(=O)NCC1CCN(C(C23CC2COC3(C)C)=O)C1 c1(C(C(=O)NC2CC2)N(C)Cc2nc(C)[nH]n2)ncccc1Cl C(=O)(C1=NOC2(CCN(C(=O)Nc3cc(Cl)c([N+](=O)[O-])cc3Cl)C2)C1)N(C)C c1(CN2C(C(=O)Nc3cncc(C)c3)CC(F)C2)cccc2ccncc12 C(CN=c1nc(N(CC(C)CN(C)C)C)c2c([nH]1)COC2)c1c(C)nn(C)c1C c1(OC)ccc(SCC(O)COc2cnccc2CBr)cc1F.C1C(=O)N1 C1(C(N2C(CNC(c3ccn(C)c3)=O)CC2)=O)Nc2ccccc2C1(C)C CC1=NOC(=O)C1CCC(=O)NCC1CCN(C(c2cc(C)n(C)c2)=O)CC1 c1(C(=O)NC2CCC(NC(c3c(OC)noc3C)=O)CC2)cnc2ccoc2c1 C12(C(N(CCCN(C(c3n(CC)ccc3)=O)C)C)=O)CCCCC1CS(=O)(=O)C2 CC(C)CC(C(=O)NC1CC(O)C1)ONC(c1ccc(F)cn1)=O Cc1c(CNC(C2CCC(NC(=O)C(O)c3ccsc3)C2)=O)cccc1F C1(C(=O)NC2CCN(C(CC)=O)CC2(C)C)CCc2nc(CC)ncc2C1 C(=O)(C(CCOCCO)NC(=O)COCCF)C1(C(C)NC(=O)C2CC2)CC1 Cc1[nH]nc(CN2CCOCC2)c1NC(c1ccccc1SC(F)(F)F)=O c1(C(N2CC(OC)(CNC(=O)C(C)(F)C(C)(C)F)C2)=O)nccn2c(C)nnc12 N1(C(C(CNC(C=C(CC)CC)=O)OC)=O)CCc2nc(O)[nH]c2C1 N1(C(c2c(C)c(Cl)cnc2)=O)C2CCC1CC(CC(C)NC(c1cnns1)=O)C2 C#CC1(O)CCN(C(C23CC2CCN3C(c2ccc(C#N)o2)=O)=O)C1 N1(C(C2(C(C)(F)F)CC2)=O)CCCC(NC(C2CCCCO2)=O)C1 Cc1cc(C(c2nnnn2C2CC(F)(F)C2)NC2CCS(=O)(=O)C2)c(C)nn1 N1(C(C(C)(N(C(CC(C(C)C)C)=O)C)C2CC2)=O)CC2(CCNC2=O)C1 C1(C(=O)NC(C(=O)NCCN(C)CCO)C2CCC2)CC2CCCC2C1 CC1CS(=O)CCN1C(=O)CC1CN(C(=O)CSC(C)(C)C)CC1F N1(C(c2ccc(CC)nc2)=O)CCC2(CC1)CC2NC(=O)Cc1ccccc1 Cc1ncc(F)c(N2CC(NC(C3(C#N)CC3)=O)C(F)C2)n1 C12(C(N3CCCC(c4cccc(OC)c4)C3)=O)CCCC(C(=O)OC)(COC1)C2 C#Cc1cc(C(=O)NC(CNC(c2nocc2C)=O)CC(C)C)ccc1C C(CC(O)C(C)C)NC(CCN(C(C(CC)O)=O)CC)=O c1(C(N(CCN(C(C(CC#C)C)=O)C)C(C)C)=O)cc(Cl)cnc1C Cc1cccc(Cl)c1C(=O)NCC1(NC(c2coc(Cl)c2)=O)CC1 N1(C(C2C(C)OCC2)=O)CCCC(C2CN(C(c3ccccc3[N+](=O)[O-])=O)C2)C1 c1(C(N2CC3C(NC(CCCSC)=O)(C3)C2)=O)ccc2c(c1)CCC2=O N1(C(c2nc(COC)sc2)=O)CC2CCC2(CNC(C2(C)CCCCO2)=O)C1 Cn1ccn2ncc(C(=O)NC3CC(NC(c4n[nH]c5c4CSCC5)=O)C3)c12 C1(c2n(C(C)C)nnn2)(NCC(C)(C)N(C)C)CCCC(S(C)(=O)=O)C1 C(=O)(C(F)(CNC(=O)C(c1ccn(C)c1)C)C(C)C)N(CCN(C(C)=O)C)C C1(CC)CN(C(c2cc(-c3ccccc3)on2)=O)CCC1Nc1ncc(F)cn1 N1(C(C(N2CCCCC2C2CC(C)CCC2O)CC)=O)CCc2c(F)cccc21 N1(C(c2cc(C)[nH]n2)=O)CC(CNC(=O)CCc2ccc(F)cc2Cl)C(C)(C)C1 C1(O)(C(C(=O)N(C)CCN(C)C2CC2)F)CN(C(=O)CC2(C#N)CC2)C1 CC(C)C(C(=O)N1CCC(C(=O)NC2CC2C(F)(F)F)(CO)C1)C1CCC1 N1(C(c2cncc(C#C)c2)=O)CCC(NC(=O)C(C)(C)SC)C(C)(C)C1 n1(CC)cc(CC(=O)NC2COCCC2NC(C2(C)CCCO2)=O)c(C)n1 CCC(C(=O)NC(C)CCNC(=O)Cc1ncc(Cl)s1)C(F)(F)F c1(CC)ccccc1.C1(COCC)CCCC1C=CC=CC(=O)NC1CC(CC)C1 N1(C(C2C(CC)CCO2)=O)CCC(C(=O)NC2CC(=O)NC2=O)(CC)C1 N1(C(CCCC=C)=O)CC2(CC)CC1(CNC(C1(F)CC1)=O)C2 c1(CC)cnc(C(=O)NC2CN(C(=O)CN(C)C(C)C)CC2n2cccn2)cn1 C(=O)(C#CC1(C)CCCO1)NCc1ccc(C(N2CCC(C#C)CC2)=O)s1 C1(C(=O)NC(c2ncco2)C)(OC)CCCOC1.C1(OCC)CCC1CNC=O C12(NC(C(C(C)NC(=O)COC3CC=CC3)(C)C)=O)CCCN(CCC1)C2 C(c1ccc(F)c(F)c1)=C(C)C(N1CC(NC(=O)C(C)CCO)CC2(CC2)C1)=O CC(C)(C)C(C(=O)NCC1CCCC1NC(C1(N(C)C)CCC1)=O)n1ccnn1 c1(C(=O)OCC)cccnc1OCC1CCC1.c1ccccc1.C12CCC1NC2=O C1(C(N2CC(NC(C3(F)CCCC3)=O)C2)=O)(CC)CCOC1 c1(C(=O)NC(CCOCC)C(=O)NCC2(C)CCC(=O)N2C)cccc(C)c1F C1(CN(C2CCC2)C(=O)OC)C2CN(C(=O)Cc3cncn3C3CC3)CC12 n1(C(C)C)nccc1C(=O)O.n12cc(nn1)CC(C1CC1)C(=O)NCC2 CCCC(C(=O)NC(C)CN(C(=O)CCn1cccn1)C)NC(=O)OC(C)(C)C C1(CNC(c2nccs2)=O)CC2(CCC2)CN1C(c1ccn(CC(F)(F)F)n1)=O CN1CC(O)CC1(C)C(=O)Nc1ccc(-c2cncc(F)c2)c(F)c1 CCCCCCCCNC(=O)C(=O)NC1CCC(NC(C2C(F)(F)C23CC3)=O)CC1 C1(C(C)C)CN(C(c2cc(C3CC3)on2)=O)CCN1C(c1cn2ccsc2n1)=O C1(C)(C(=O)NCCN(C(c2cccc(OCC)c2)=O)CC)CCCNS1(=O)=O c1(C(C)NC(=O)CC#N)c(F)cccc1Cl.n12cc(nn1)CC1(O)CN(C1)C2=O CCC(CNC(C1(F)CC1)=O)(CC)NC(c1ccc(C2CC2(Cl)Cl)cc1)=O c1(C(=O)NC2CC(C)N(C(=O)CC(=O)N(C)C)CC2)cccc2c1CCC2 C1(NC(C(C)OCCOCC)=O)CCC(CC(=O)NC2CSC2)C1 C(=O)(C(C(C)C)c1cnn(C)c1)N1CC(C)(NC(COCC(C)C)=O)C1 C1(NC(CCn2ncc(C)c2)=O)CC2CCC1N2C(C1CC12CCSCC2)=O c1(C(N(CCCCNC(C=C2CCN(C)C2)=O)C)=O)cccc(CF)c1 C1(CC)CCN(C(c2cnc(O)o2)=O)C1C(=O)N(C1CC2(CC2)C1)C C(CCC(=O)NC1C2CCN(C2)C1=O)=CC.c1(CC)nncn1CC C1(F)(C(=O)NCC(C#C)(C)C)CCN(C(C2(C)CCC3CC3C2)=O)CC1 C(=O)(CC(C(=O)N1CCCC1(C)CNC(c1cccc(C)c1)=O)N(C)C)OC N1(CC2OCC(C)(C)C2)CCC2(CC1)CC2(C)C(N1CCNC(=O)C1CCO)=O C=C(C)CC(C(=O)O)NC(=O)CSCc1cn(-c2ccc(Cl)cn2)nn1 c1(C(N2C(C)(C(=O)NC(C(=O)NC)C)CC2)=O)c(F)cc(Br)cc1F N1(C(CC)=O)CCCCC1C(=O)NC(=O)Cn1cc(CNC2(CC)COC2)nn1 N1(C(C(C)(C)n2cnnn2)=O)CCCCC(C(N2CCC(C(F)F)CC2)=O)C1 C=C(C)C(C)(O)C(=O)NCC(C)(C)NC(=O)C(C1CCCC1)OC c1(CNC(=O)NCCc2ccc(C3CC3)nc2)nc2ccccc2n1C(F)F c1(C(=O)NCC(C)(C2CC2)NC(c2c(OC)nsc2)=O)cc(C)cc2c1CCC2 C1(C(=O)NC2(C(=O)NCC)CC2)CC2(CCC2)CN1C(=O)C(C)(F)C(=O)OC N1(C(CC(=O)NCC)=O)CC2CN(C(=O)C(C)Sc3ccccc3)CC2C1 n1(CC2CC(C)C2)nc(-c2cccc(Br)n2)nc1-c1cn(C(C)(C)C)nn1 c1(C(=O)NCCC2(CNC(C(C)C#N)=O)CC2)cc(O)nc(O)n1 C(=O)(CCS(=O)(=O)CC(C)C)N(C1CCCN(C(C(CC)CO)=O)C1)C c1(C(=O)NC2CCCCN(C(C(C)(C)CC3CC3)=O)C2)ccc([N+](=O)[O-])cn1 C(=O)(C(C)(C)N(C)C)NCCN(CCOC)C(c1ccnn1C1CC1(F)F)=O CCC(C)(CCNC(c1cccn1C)=O)NC(=O)C(C)N1CCCC1 C1(C(N2CC3(N(C(CC(C(C)C)C)=O)CC3)C2)=O)CCC2(CC1)CC2(F)F N1(C(C2CC(OC)C2)=O)CCOCC1CNC(c1ccnc(C(N)=O)c1)=O c1(CCC(=O)NCCNC(C)=O)nccn1C.C1(=O)C(=O)N(CC)CC(C)N1 Cc1cc2cc(NC(C3CC3NC(c3cc(C)n(C)n3)=O)=O)ccc2[nH]1 C(=O)(CCCCC(=O)NCC(=O)NCc1ccc(Br)c(F)n1)NC CC(CCCc1ccccc1)C(=O)NCC1CC1NC(c1ccc(CC2CC2)s1)=O S(=O)(=O)(CC(=O)N1CC2CC2(CNC(=O)CCC2CCCCC2)C1)N(C)C Cc1ccc(C(=O)NCC(C2CCCN2C(C2CCC(C)CC2)=O)(C)C)cc1C C1(CC(N2CC3CCN(C(C(C(=C)Cl)(C)C)=O)CC32)=O)CCc2sccc2C1=O N1(C(c2cc(C(=O)OCC)n(C)n2)=O)CCC(NC(c2coc(Cl)n2)=O)C(C)C1 N1(C(C)CC2(C)CC2)CCC2(CC1)CC2C(N1CCCCCCC1C)=O n1(CCC)ncc(C(=O)NC(C)(CNC(C2CCCCC2O)=O)C(C)C)c1C N1(C(C(C2(O)CN(C(C3N(C)CC(F)C3)=O)C2)F)=O)Cc2n[nH]cc2C1CO C1(NC(C(C)c2cncs2)=O)CCC2(CCN(C(=O)C(c3ccn(C)n3)C)C2)C1 c1(C(=O)NCCC(C)NC(c2nc[nH]c3nccc2-3)=O)ccnc2[nH]c(O)nc12 C=CCC(CNC(c1cscc1C1CC1)=O)C(=O)N1CCC(NC(=O)OCC)C1 c1(C(N(CCCCNC(=O)CCC2CC2(F)F)C)=O)ncc2[nH]ncc2n1 c1(C(N(C2CCC(NC(C(C)n3cnnn3)=O)CC2)C)=O)ccc(O)c(N)c1 C1(C(=O)NC(CN(C(Cn2c(C)nnn2)=O)C)C)CCCCC1c1cccnc1 C(=O)(C(C1=NOC2COCC12)N(C)Cc1c(F)cc(F)cc1F)NC(C)C c1(N(C(CCSCC)C)C)nc2c(c(=NCCNc3ccccc3Cl)[nH]1)COC2 C1(C(N2CCOC(c3ccccc3)C2)=O)CC(F)CN1Cc1nccs1 c1(OC)cnc(C(=O)N(C2CCC(NC(c3nnc(C(C)(C)C)s3)=O)C2)C)cn1 Cc1cc(C#N)ccc1-c1csc(C(=O)Nc2c(C(N)=O)cnn2C)c1 C1(C(=O)OCC(CC)NC(C2CC2)C)CC2CCC1CC2 Cc1cc(C(=O)NC2CCC(CC(=O)NCC3CCCO3)CC2)ccc1C#N Cc1ccc(C(=O)N(CCCCC(=O)NOCC2CC2)C2CC2)cc1C#N Cc1cc(C(=O)NCCOCC(=O)N(C2CCCC(C)C2C)C)nnc1C N1(C(c2c(C)oc(Cl)n2)=O)C2CCC1CC(CNC(=O)C(C1CCCCC1)O)C2 N1(C(C2Cc3cc(F)ccc3O2)=O)CCCC(C2CCNC2)C1 Cc1c(F)ccc2[nH]c(C(N3CC(C(N)=O)(CNC(=O)CSC)C3)=O)cc12 c1(C(=O)NCC2C(C)CCC2)cccc([N+](=O)[O-])c1Br C1(N(C)C)CCCC(C(N2CCC(O)(n3cc(C(C)(C)S(C)(=O)=O)nn3)C2)=O)C1 CC1CC=CCC1NC(C1(CO)CCN(C(c2cccc[n+]2[O-])=O)C1)=O C1(CNC(CC(=O)NC)=O)CCCC12CN(C(c1c(C)cc(Br)cc1Cl)=O)C2 c1(C(N2CCN(Cc3c(Cl)ccnc3Br)CC2)=O)ccc2occc2c1 c1(C(N2CC3(C(=O)OC)CC2CO3)C(=O)NC)cc2ncccc2o1.C1CCN1 c1(CNC(c2nnnn2CC(F)F)(CSC)C)ccc(OC)c(C(C)C)c1 Cc1cc(F)c(C(=O)NC2CN(C(C3CCc4ncnn4C3)=O)C2)cc1Br CC1C(NC(=O)CC2CCC(=O)NC2=O)CCCN1C(c1cc2n(c1)CCC2)=O C(=O)(C(C(C)O)NCC(C)C)NCCC(C)C.C1C(C)(C)OC2(CC2)C(=O)N1C c1(CNC(C2(c3ccccc3)C(C)(C)C2)=O)ccc2nccn2c1 Cc1cnc2c(C(=O)NCCCNC(C3CCCC(F)(F)CC3)=O)cccc2n1 N1(C(C2CC(C#N)C2)=O)CCN(C(c2ccc(CC#N)c(Br)c2)=O)C2CC12 c1(CCC)nc(C)c(C(=O)NCCOCCN(C)C(c2c[nH]nc2F)=O)s1 CCCCC(F)C(=O)NC(C)CC(=O)NC1CCOC(C)(C)C1 C=CCCC(C(=O)NCCn1ccnn1)NC(c1coc(SC)c1)=O CC1CCCC(C)CN1C(c1coc(CNC(=O)CC=CC(C)(C)C)c1)=O c1(C(C)C(=O)NC(CNC(=O)Cc2nccn2C)C2CC2)ccc(Cl)cc1 C1(NC(=O)CCC2CCCCO2)C2CN(C(=O)CC3CC(F)(F)C3)CC12 CC(CCNC(c1n[nH]cc1F)=O)CCNC(c1cc(-c2ccccc2)no1)=O C=CC(C)(O)C(=O)NC(C1CCN(C(=O)C(C)COc2ccccc2)C1)C CC1(C)C(NC(c2n[nH]c(=N)[nH]2)=O)CC1CC(N1CC(n2cccn2)C1)=O C1(C)(CNC(c2c(CC)n(C)nc2)=O)CN(C(c2nc(Cl)sc2C)=O)CC1C C1(CC(=O)NC(CNC(C(C)NC(CC)=O)=O)(C)C2CC2)CCCC(C)(C)O1 N1(C(C(C)=CC)=O)CCC2(CNC(=O)CCCN3CCCC3)CCCCC12 C(=O)(C(CC(C)(C)C)OC)N1C(CCC)CN(C(=O)CCC2CCCC2)CC1 c1(C(=O)NCC2CN(C(CCSCC(C)C)=O)C(C)CC2)cc2c(s1)CCC2=O c1(N2CC(C(CC)NC(c3c(S(C)=O)cccc3)=O)C2)nc2ccc([N+](=O)[O-])cc2s1 c1(C(N(CCF)CC)=O)ccc2c(n1)CN(C(C1CCC(C)(C)CC1)=O)CC2 CC(C(C)(C)C(=O)NCC1(O)CCC1)NC(=O)C(c1ccccc1)F N1(C(C(CC)(C)O)=O)CCC(C2CCN(C(c3ccc(C(C)C)s3)=O)CC2)CC1 c1(OCCCCC)ccc(C(=O)NCC(C2CC2)NC(=O)CS(N)(=O)=O)cc1 CCC(CC(=O)N1CC(OC)CC1CNC(=O)COCC(F)F)OC c1(C(C)C)ccc(C(O)C(N2CCC(OCCNC(C3CCSC3)=O)C2)=O)cc1 C1(O)(C(=O)NCCCCCN(C(C=NOC)=O)C)CCCC(C)(C)C1 C=CCC(C(=O)NCC#CC(=O)N1CC(CO)(CO)C1)OC c1(C(N(CCCNC(C2C(C)CC2)=O)C2CC2)=O)cc(O)cc(Cl)c1 C1(C(c2n(C3(C)CC3)nnn2)NCC2CC(c3ccccc3)C2)CCCCC1C c1(C(=O)NC2C(CC(C)(C)C)C2)ccc2c(n1)CN(C(=O)CCCF)CC2 C1(C(N(CC(F)(F)F)C(C)C)=O)CCCC(n2cc(-c3cnsc3)nn2)C1 Cc1ccccc1NC(=O)C(c1csc(Br)c1)N(CC(=O)N(C)C)C CN1CC=C(CC(=O)N2CC(NC(C3CCC(C(N)=O)C3)=O)CC23CCC3)CC1 C1(CN=c2cc(COC)nc[nH]2)CN(C(c2ocnc2C)=O)CC12CCOCC2 N1(C(CC(CNC(CN2CCN(C)CC2)=O)O)=O)CCCC2(CC1)CC2 c1(C(N(C2CCCN(C(C3(CSC)CCOCC3)=O)C2)C)=O)cc(Cl)cnc1O c1(C(C(=O)NCC(C)C)N(C)CC2CC2(C)C)ccc2ccn(C)c2c1 N1(CC(N2CC(CC(C)NC(c3c(C)nncc3)=O)C2)=O)CCc2ccccc21 c1(C2(CN3CC(C(O)CF)C3)CCC2)ccc(OC(F)(F)F)c(Cl)c1 C1(=CC(=O)NCC(C(=O)NCC(C#C)CC2CC2)N(C)C)CCC(C)CC1 C(=O)(CC(C(N)=O)c1ccccc1)C1(C)CC1.C(C(C)C)c1nnnn1C C1(C)(C(N2CC(C(C)NC(=O)CNC(=O)C(C)(C)C)C2)=O)CCCC1C C1(O)(CC(=O)NC2CC(O)(CNC(=O)C(O)C3CCCC3)C2)CCCC1 Cc1cc(C(=O)NC2CN(C(=O)COCC3CC3)C(C)(C)C2)cc2nn[nH]c12 C1(N(C(=O)Cn2cc(C3CC3)nn2)C)CN(C(=O)Cc2ccc(Cl)cc2)CC1(C)C Cn1cnc(C(=O)NCC2(C(N3CC(O)(CO)C3)=O)CCCO2)n1 N1(C(CC2(C=C)CCCCC2)=O)CC2CCC(C1)N2C(=O)COC1CCOCC1 c1(C(=O)OC)cccc(Nc2cc(SC(=O)C(C)(C)C)nc(C)n2)c1C C1(CCC)CN(C(=O)NCC(N2CCN(CCOC)CC2)=O)CCO1 N1(C(c2cccnc2Cl)=O)CC(C2CCN(C(C3(C(F)F)CC(O)C3)=O)CC2)C1 N1(C(C2CC(OC)CN2C(c2cnc(O)o2)=O)=O)CCc2nc(O)[nH]c2C1 C1(C(=O)NCC=CC2CC2)CC(C2CCOCC2)=NO1 C1(OC)C(NC(C2(F)CCN(C(C3(CC4CC4)CCC3)=O)CC2)=O)CC12CCC2 N1(C(C2(F)CCN(C(c3c(C)n[nH]c3C)=O)C2)=O)Cc2c(O)n[nH]c2C(F)(F)C1 CN1CCCC(C(N2CCC(C(=O)NCc3cc(C4CC4)no3)C2)=O)C1 C1(C(=O)NCC(C(=O)NCCc2cn(CC)nc2)C)CC(=O)CCO1 C1(NC(CCCCC)=O)COC2(CCN(C(c3ocnc3C(F)(F)F)=O)C2)C1 C1(Nc2cn(CC)nc2)(CO)CCN(C(C2(C)CCNC2=O)=O)C1 C(=O)(C(C(C1CC1)OC)N1CCC(OCC)CC1)NCCCC C1(CN(C(Cc2cc(C)[nH]n2)=O)C)CCCC(NC(C2(C)CCCC2)=O)C1 N1(C(C(CC)CC)=O)CC(NC(=O)CCC2CCCCN2C(C)=O)C(C)(C)C1 C(=O)(C(CNC(c1cnnc(O)c1)=O)CC1CC1)NCC(C)CC1CC1 c1(C(=O)NCC2N(C(C3CN(C(C)=O)C3)=O)CC2)csc(C(N)=O)n1 C1(C(N(CCN(C(C)C)C(c2sccc2OC(F)F)=O)C)=O)CC2CC1CO2 N1(C(=O)CCc2cn(-c3ccnc(Br)c3)nn2)CCc2nc[nH]c2C12CCNC2 C1(C)(CC(C)C)CCCN1C(=O)COC1CN(C(=O)C(c2cnn(C)c2)C)C1 c1(C(=O)NCC2N(C(COCCCCCC)=O)CCCC2)cc2ncccn2n1 c1(C(=O)OCC(C2C(C)(C)C2)=O)nccn1O C(=O)(CCCCCOCC)NC12CC(NC(C(C(=O)OCC)C3CC3)=O)(C1)C2 c1(CNC(C2CC2C(=O)NC2(c3ccccc3)CC2)=O)ccc(Cl)cc1Cl C1(NC(C(C)=C(C)C)=O)CCN(C(C2CCC(C)(C)O2)=O)CC1C N1(C(C(CCSC)NC(c2cccnc2)=O)=O)CCC(F)(F)CC1C N1(C(C(C)C2(O)CCC2)=O)CC(C)(C)CC1C(=O)NCCOC1CCCC1 N1(C(C(CC=CC)C)=O)CC2CCN(C(=O)CC3(CC)CCC3)CC(C2)C1 C(=O)(C(F)(F)C(O)C1CC1)NC1C2(CC(NC(c3ccccn3)=O)C2)C1 c1(C(N2CC(NC(c3c(OC)n[nH]c3)=O)C(CO)CC2)=O)cccc2ncsc12 c1(C(N2C(C)(CNC(CC(C)OC)=O)CCC2)=O)cc(C)nc(Cl)c1 C1(C(=O)NC2CC(CNC(C(C)Sc3ccccc3)=O)C2)CC2CC2CC1C C(=O)(C1=CCC(C)CC1)N1CCC(C)(NC(COCCCOC)=O)C1 N1(C(CCCCC#C)=O)C2CCC1CC(CCNC(=O)C(C1CCCCC1)O)C2 c1(CCNC(C)=O)cc(C(N2CCCC2C2CCCCC2)=O)no1 Cc1cc(C(=O)NCC(=O)NC(C)CCCNC(=O)Cc2nc(C)cs2)cc(C)c1 N1(C(c2ccc(C#C)cc2F)=O)CC2CCN(C(=O)CCC3CCOC3)CC2C1 N1(C(C(CC=C)CNC(c2cc(Cl)ns2)=O)=O)CC2CC(C1)C2(C)C c1(NC(=O)CC2CC(Cn3cc(Br)cn3)C2)cccc(COc2ncccn2)c1 c1(NC(CN(c2ccccc2)CC(=O)OC)=O)cc(C(=O)O)cc(Cl)c1 C#CCCC(=O)N(C(CNC(c1cn(Cc2noc(C)n2)nn1)=O)C1CC1)C CC(CCNC(C1(C)CN(C(=O)C(C2CCOCC2)=O)C1)=O)CC(C)(C)C C(=O)(CC1COc2cccc(Br)c21)NC(CC#C)CO C(CC(C)C)(C(N)=O)NC(CC1C2CN(C(C3N(C(C)=O)CCC3)=O)CC21)=O c1(C(=O)NCC(CNC(c2sc(=N)[nH]c2C)=O)OC)nnc(C)cc1O CCCCC(C)C(=O)NCC1(COC)CCCN1C(=O)C(F)CC1CC1 C1(C)(C(=O)NC(C2CN(C(C(CC=C)NC(C)=O)=O)C2)C)CCC(F)(F)C1 O=C(C1CCc2cccc(F)c21)NC1CCCN(C(=O)CC2CC2)CCC1 c1(Cn2c(-c3cncc(OC)n3)nc(COC)n2)ccc2ccccc2n1 c1(C(N2CC(NC(CCOC)=O)C(F)CC2)=O)cc(F)c(F)c(Br)c1F c1(NC(CC(=C)Br)=O)cc(C)nc(O)n1.C12CCN(CC1)C(=O)c1cn2nn1 C1(C(N2CC(C)(CCC(=O)NC(c3c(C)nns3)C)C2)=O)CCC(=O)N1C C1(C#N)(C(N2CC(OCCNC(c3cnc(COC)s3)=O)C2)=O)CCCCC1 N1(C(Cc2ccc(C#C)cc2)=O)CC(CNC(=O)C=CC(C)C)OC(C)(C)C1 c1(OCC)cccc(C(N2CC(F)(CNC(C3CC4CC34)=O)C2)=O)c1 c1(C(=O)NCC2CN(C(COCC=C)=O)CC2O)cnc2ccccc2n1 c1(CNC(C=C2CCN(C)C2)=O)ncccc1CNC(C1(c2ccno2)CC1)=O C(=O)(CP(=O)(C(C)C)C(C)C)NCC1C(NC(c2ccc(C)c(N)c2)=O)CCC1 C1(C(=O)OC(C)C)OC(C)(C)OC1CNC(=O)NCC1COC(C)(C)O1 c1(CC(=O)NC(CNC(CSCCOC)=O)C(C)(C)C)cn2c(n1)CCCC2 c1(C(=O)NC2C(NC(c3c(COC)nn[nH]3)=O)CCC2)ccc(F)c(F)c1F N1(C(CC2C(C)OCC2)=O)CCN(C2CN(C(=O)CC3CCOC3)C2)CC1 C(=O)(C1=CC2CC(C1)CC2O)NC(C)CCCNC(c1c(N)cccc1F)=O Cc1cc(NC(C2CC(F)CN2Cc2ccc(Br)cc2I)=O)cc(Cl)n1 c1(N(C2CN(C(C3(C)C=CCC3)=O)C2)C)nc(Cl)nc2c1SCC2 C=CCCCCCC(=O)N(CCCCNC(c1cc(C)cnc1C)=O)C Cc1cnc(C(=O)NC2CCC(NC(c3cn(CC(N)=O)nn3)=O)CC2)cc1C c1(NC(CCNC(C(CCSC)O)=O)C)nc(C)nc(O)c1C C(=O)(CC1CCc2ccccc21)NC1C2CN(C(c3cnc(C)s3)=O)C(C2)CC1 Cc1c(C(N2CC3CC2CN3C(=O)CC2=NNC(=O)C2)=O)cc(N)cc1O N1(c2c(C)c(NCc3cc(F)cnc3Cl)ncn2)CCC2(CC1)CCC2(C)C c1(C(=O)NC(Cc2cc[nH]n2)C(=O)NCCCN2CCC2)ccc(F)cc1 C1(CCNC(C(n2ncc(C)c2)C)=O)CSCCN1C(=O)CSC(F)F c1(OCC#C)ccc(C(=O)NC(C)CCNC(=O)C=Cc2cscn2)cc1 N(C1c2ccccc2OCC1O)C(=O)NC1C(c2ccc(C)cc2)OCCC1 Cc1ccc(O)c(CNC(C2C=CCN(C(C3COCCC3C)=O)C2)=O)c1 CC(C)(C)CC(C)(C)C(=O)NC1CC(F)(CNC(=O)CCCC(N)=O)C1 N1(C(c2c(C#C)cnn2C)=O)CCN(C(c2ncsc2C2CC2)=O)CC12CC2 N1(C(c2cnn(CC)c2C)=O)CCN(C(c2ncc3ccccn23)=O)C(C)C1C C1(CNC(C(c2cccnc2)C)=O)CC(C)N(C(=O)CC2OCCC2(C)C)C1 C1(NC(C(C)NC=O)=O)C2CCN(C(=O)CC3CCC(C)C3)CC12 C1(CCNC(c2cnc(O)s2)=O)CN(C(=O)CC23CCCC2C3)CCS1(=O)=O C1(N(C(=O)CCc2ccc[nH]2)C2C(c3cn(C)nc3)C2)CC2CC1CN2 Cc1nccc(C(=O)NCC(CC2CC2)C(=O)N(C)CCC2CCCC2)n1 C=C(C)CCN=c1[nH]c2c(c(=NCCCCC3CC3C)[nH]1)COC2 N1(C(c2nc(SC)sc2)=O)CCCC2(CCCCC2NC(=O)Cn2ccnn2)C1 C1(CNC(CC2(CSC)CC2)=O)CCN(C(=O)CCCc2ccccc2)CC1O CC(C)C(O)C(C)C(=O)NC1(C(=O)NCC2CCCCS2)CCCCC1 c1(C(CCOc2ccc(Br)cc2)NCc2n(CC)ncc2)cccc(C#N)c1 C1(NC(C(c2cc(F)cc(F)c2)(C)C)=O)CCCCN(C(C2CCCCO2)=O)C1 N1(C(c2c(C)cno2)=O)CC2C(NC(=O)C(c3cccc(Br)c3)C)C2C1 CON1CCC(c2nnnn2C2CCC2)(NCC2(C(C)(F)F)CC2)CC1 c1(NC(CCNCC(CCCC)CC)=O)cc(=NC(C)CS(C)(=O)=O)[nH]c(C)n1 c1(NCCC2CCCN(C(Cc3c(C)nn(C)c3)=O)C2)ncnc2cc(Br)sc12 C(C(CC1CC1)C(=O)N1CC(c2ccccn2)C1)NC(=O)C(Cl)=CCl C=CC1CCCN1C(=O)C(C1(O)CCCCC1)NC(=O)CN(C1CCC1)C C=C(C)CCC(=O)NCC(CC(C)C)NC(=O)C(F)CC1CCCCC1 c1(CC)cc(C(=O)NC(C)C(C)NC(c2ccccc2CO)=O)cc(C)c1 C=CCC(CNC(C1CC(C)=NO1)=O)C(=O)NC(CC)CO c1(C(N(c2ccn3ncc(Br)c3n2)C2CC(N)C2)=O)[nH]c2ccccc2c1Cl C1(C(=O)NCC(C)NC(c2cn(C)nc2C(F)(F)F)=O)Cc2ccccc2N1C Cc1cc(C)c(C(=O)NCC(O)CNC(C2(O)COC2)=O)cc1N N1(C(C2C(C)C2(F)F)=O)CC2(C1)CN(C(=O)CCC1CCCCO1)C2 C1(NC(CNC(CC)=O)=O)CC2CCCC(C1)N2C(=O)CC1CCCCO1 CCCCCC(C)CC(=O)NC1CCN(Cc2ccc(Cl)cc2C)CC1 C(=O)(C1c2ccnn2CCN1C(=O)OC(C)(C)C)Nc1c(C)nn(CC(F)(F)F)c1 c1(CC)cc(C(=O)NC2(CC(=O)NCc3cscc3Br)CCC2)ccn1 c1(CN(CC(=O)NC(CCN(C(C(C)=CC2CC2)=O)C)C)C)ccc(C)cc1 CC1(NC(C2C=CCS2)=O)CCCC1NC(c1cncc(F)c1)=O c1(C(=O)NCC2CCCN2C(=O)C=CC2CC2)cccc(F)c1O N1(C(c2ccc(CC)o2)=O)CC(NC(c2cncn2C)=O)C(C2CC2)C1 C12(C(N(CC(CN(C(C(C)N(C(C)=O)C)=O)C)O)C)=O)CC(C1)S(=O)(=O)C2 NC(=O)N=Nc1ccc(C(=O)NCc2[nH]ccc(=O)c2O)cc1 N1(C(C(CC#C)O)=O)CC2(CCCCN2C(c2ncc(Cl)cc2F)=O)C1 Cc1nc2cc(C(N3CCCC3Cc3ccsc3)=O)ccc2n1C(C)C Cc1cc(CC(=O)NCC2(C)CCCN2C(=O)C(C)Cc2cnc[nH]2)cc(C)c1 C=C1CC(C)(NC(=O)C(O)C2CN(C(C3CCCN3CCC)=O)C2)C1 C1(C)(CC)C=C(C(=O)NC2CC(F)(CNC(c3cnccc3C)=O)C2)C1 n1(CC(=O)NCC2(NC(C(c3ccnn3C)C)=O)CCC2)nnc(=N)[nH]1 c1(OC)cc(CC(=O)NCC(C)NC(C2CCO2)=O)ccc1C c1(C(=O)NCC2N(C(CC(=C=C)C)=O)CC2)cc2cc(Cl)c(Cl)cc2[nH]1 c1(C(=O)NC2CCNCC2(F)F)nn2c(c1Cl)OCCC2 Cc1ccc(C(=O)N(C2CC(NC(c3cnc(O)s3)=O)C2)C)c(C)c1 C12(CNC(c3n(C)cnc3)=O)CCC(CN(C(C3(C)CC3(Cl)Cl)=O)C1)C2 C(=O)(C1=NOC2COCC12)NC1(C)C(C(=O)NCCCCC#C)CCCC1 C1(NC(c2ccc(Cl)c(Cl)c2)=O)CC2(C1)CC(NC(c1cc(Cl)cnc1F)=O)C2 c1(C(N2C(CN(C)C(C3CCC(=O)C3)=O)CCC2)=O)ccc2nsnc2c1 N1(C(c2c(C)ocn2)=O)CCN(Cc2cccc(Br)n2)CC1CC#N Cc1cc(N2CCCC(CNc3ncccn3)C2)nc(N(CC(F)F)C)n1 C1(CNC(C(C)OCC#C)=O)CC2(CO1)CN(C(=O)C(C)=C1CCCC1)C2 CCC(C)CC(=O)NC1CCC1NC(C1(Oc2ccccc2F)CC1)=O CC1(Cc2cn(C)nn2)CCCCC1(F)F.C(C(=O)NOCC1(O)CCC1)O c1(C(N2CC(NC(CCCCCOC)=O)C(C)CC2)=O)cc2c(cn1)CCCC2 Cc1cccc(C(=O)NC2(C3CC3)CCC2)c1.C1C(C)C(=O)N1 c1(CC)cc(OC)ccc1NC(=O)C(N1CCCC(OC2CCCCC2)C1)C c1(C(N(C(CCNC(CCN(CCCCC)C)=O)C)C)=O)cc(O)ccc1Cl CC1(CNC(c2ccnc3ccccc23)=O)CCC(O)CC1C(=O)O N1(C(C)=O)CCCN(C(C2(CF)CCN(C(=O)C3CC3)C2)=O)CC1 Cc1ncc(C(=O)NCC2(C)CC(NC(=O)CSCC(F)F)C2)cn1 C(=O)(C(F)CC(C)(C)C)N1C(C)CCC(C(=O)Nc2c(C)ccnc2)C1 C1(C(=O)NCC2(OC)CC2)CC2CC1CC2NC(=O)C(C1CCOCC1)C C1(CNC(c2c(CC)nc[nH]2)=O)CC(C(C)C)CCN1C(=O)C(C)COC c1(CC)ccccc1-n1cc(-c2ccccc2NC2(C(=O)O)CCC(C)C2)nn1 C1(NC(=O)CC23CCCC2C3)CCCCC12CCCC2 c1(-c2n(CC)c(N3CCC(OCCO)CC3C)nn2)cnccc1C#N N1(C(c2c(CC)con2)=O)CCC(C2CCCN(C(=O)C3=C(Cl)CC3)C2)C1 C1(C)(NC(CC)=O)CCCCC1C(=O)N(CC(C)SC)C C(CCC(C(=O)NCC1(CO)CC=CC1)NC(C1CCC(C)(O)CC1)=O)OC N1(C(CC2N(C)CCOC2)=O)CCC(NC(=O)CCc2nc(O)n[nH]2)C(F)C1 C1(C2(O)CN(C(C3CCC(OC)CC3)=O)C2)(CNC(CNC(CCC)=O)=O)CC1 N1(c2c(C(=O)OC)cccn2)CCC(NC(=O)CCCNC(N)=O)C(CO)CC1 c1(C(N2CCC(C)(NC(C(C)CC(N)=O)=O)C2)=O)cn2cc[nH]c(=O)c2n1 CC(C)CC(=O)NNC(=O)C(C)OC(=O)CCN1C(C)CCC1C N(C1CCCc2nc[nH]c21)C(N1CCCCCCC1)=O C(CCC(C)NC(=O)NC(C)C(F)(F)F)OC C(=O)(C(C)CC(=O)N1CCN(C(c2ccc(F)nc2)=O)C(C)C1)OC c1(C(=O)NC(CN(C)C(C2CCC(C)(C)CC2)=O)(C)C)ccc2c(c1)OCCN2 Cc1cc(C(=O)N(C)CCN(C(=O)CC2CCCC23CC3)C)sc1C CC1CN(C(c2ccoc2)=O)CCN1C(c1cn(CC2CNC(=O)O2)nn1)=O N1(C(=O)C(F)C2CC2)CC2COCC2(C(N2CCN(c3ccccc3)CC2)=O)C1 c1(C(N2CCC(C)CC2CNC(=O)CCCNC(N)=O)=O)ncn2c1CCCC2 C(N=c1[nH]cc2ncnc-2[nH]1)C1CCN(C(c2cc(SCC)oc2C)=O)C1 c1(OC)cccc2ncnc(NC(C)CCNC(C3CCOC(C(C)C)C3)=O)c12 c1(C(=O)NC2C(NC(=O)CC3CC=CCC3)CC2)ccc(F)c2cccnc12 c1(C(=O)NCC2CCCN(C(C=C(C)C)=O)C2)ncnc2c1CCC2 C1(NC(C(CN(C)C)NC(C2CC3COCC3C2)=O)=O)CCn2ncnc2C1 C(C)(c1ccccc1)=CC(=O)NCC1(NC(C(Cc2ccccc2)OC)=O)CC1 c1(NC(C2CCC(CC(=O)NC(C)CCO)C2)=O)cccc(C(=O)NCCC)c1 c1(NC(=O)Cc2cc(Br)sc2Br)nc2c(s1)CC(F)(F)CC2 C12(C(=O)NCC(CNC(c3ccccc3)=O)F)CCC(O)C1CC2 C1(C(N(CCCNC(c2ccc(C)s2)=O)CC)=O)C2CC1(c1cccnc1)CO2 c1(CC)nc(C(=O)NC2(CCNC(=O)C(C)CF)CC2)co1 CCCCC(C)C(=O)NCC(C)(F)CNC(c1ccnc(N(C)C)c1)=O C1(C(=O)NC2CCCC(OC)C2)CC(F)CCN1C(=O)CCC(C)(C)C c1(CC)[nH]nc(C(N2CCC(CCN(C)C(c3coc(O)n3)=O)CC2)=O)c1Cl CC1CSCCN1C(c1ccnc(CNC(=O)C2=CCSC2)c1)=O c1(CCC(N2CCC(C)(NC(c3ccon3)=O)C2)=O)ccc(Cl)c(F)c1 C(=O)(C(C)(C)CC(F)(F)F)N1CCC(c2cn(C(CCCCCC)CC)nn2)C1 N1(C(C2CCS(=O)(=O)C2)=O)CC(C2CN(C(C3CC4(C3)CC43CC3)=O)C2)C1 S(=O)(=O)(CCC(=O)NC(CNC(c1ccc(OC)cc1C(F)F)=O)C(C)C)NC Cc1cccc(-c2nc(N3CCCC(CCC4CCSC4)C3)n[nH]2)n1 c1(C(N2CC(CC=C)(NC(c3ccccc3C3CC3)=O)C2)=O)ccnc(C)c1O c1(C(N)=O)ncn(CC(=O)NC2CC(NC(=O)CCCOC(F)F)C2)n1 c1(CC(=O)NC2CC3CCC(C2)N3C(C2CC2(F)F)=O)c[nH]c2cccc(Br)c12 C1(C(=O)NC(C(=O)NC)CC(C)C)CC2CCC(C1)N2C(=O)CCC1CCC1 C1(NC(C(c2ccco2)NC(=O)CC2CCSCC2)=O)CCOCC1F N1(C(C(C2CCN(C(c3cnc(C)nc3)=O)CC2)C)=O)CCC(CO)C(C)C1 C#Cc1cnc(C(N2C(C(=O)NCC#CCOC)CCC2C2CC2)=O)c(C)c1 c1(C(=O)NC2C(CO)CCN(C(CCC(CC)C)=O)C2)cnc2c(ccn2C)c1 C(=O)(C(F)(F)CO)NCCC1CC(NC(C2(C(=O)NC)CCC2)=O)C1 C1(NC(c2cn(CC)nn2)=O)CC1C1CCCN(C(=O)C(O)Cc2cnc[nH]2)C1 N1(C(c2c3ncc(C)cn3nc2)=O)CCCCC2(CCN(C(=O)CSC(C)C)C2)C1 c1(C(=O)NC2C(CNC(=O)C=C3CCCCC3)C2)cc(Br)c(F)c(F)c1F Cc1nn(C)cc1C1=NOC(C(=O)NC2CCN(C(=O)C(C)C3CCC3)CC2)C1 C(N=c1ccnc(NC2CCC(P(C)(C)=O)C2)[nH]1)c1nc(CC)sc1 CCC(CC(C)C)C(=O)N(CCNC(=O)C(C(C)(C)C)N1CCOC1=O)CC C(CCCC(C(=O)Nc1ccc(F)cc1)N(C1C2CCCC12)C)(OC)OC c1(C(=O)NCC2CC3CC3N2C(=O)Cc2ccccc2O)cc(Cl)ccn1 C=CC1CCN(C(C2CC23CCN(C(c2cnc(C)nc2C)=O)C3)=O)CC1 c1(CN(C)C(c2cccc(O)c2)=O)ccccc1CS(N1CCC(O)C1)(=O)=O CCC(C)(CC)C(=O)NC1CCN(C(c2ncoc2-c2ccccc2)=O)C(C)C1 N1(C(CCCC)C(=O)NC2CC(C)(C(=O)O)C2)C(=O)c2ccccc2C1=O N1(C(C(CC)N(C)C)=O)CCC(C(=O)NCC(CC2CC2)OC)=C(F)C1 C1(C)(CC)NC(=O)N(CC(=O)NC2(C3CN(C(=O)CCC4(C)CC4)C3)CC2)C1=O N1(C(c2cnc(C(C)(C)C)[nH]2)=O)CCC(C2CC2)(CNC(C2CCCOC2)=O)C1 O=C(N=c1ccn(C2CCCCO2)[nH]1)Nc1ccccc1-c1cnnc(I)c1 C1(NC(C2CC3CC3C2)=O)CN(C(c2cncnc2)=O)CC12CCS(=O)(=O)CC2 CN1CCN(CC(=O)OC2(C(=O)NOCCCN=[N+]=[N-])CCN(C)C2)CC1 C(=O)(CS(=O)C(F)(F)F)C(=O)CC12CCCC1C2.C1(N)CC2(C1)CC(N)C2 N1(C(C2CCCCN2C(c2ccc(Cl)cc2)=O)=O)CC23CCC2(COC3)C1 CC1(CS(C)(=O)=O)CN(C(C2CC(CC(F)(F)F)C2)=O)C1 n1(CC(=O)N(C(C)CNC(C2CCCN(C)C2)=O)C)nc(C2CC2)n(C)c1=O c1(C(=O)NCCC2N(C(CCSCC)=O)CCOC2)sc([N+](=O)[O-])cc1Cl C(N=c1cc(C(=O)OC)nc[nH]1)C1CC(NC(c2cn(SCC)nc2)=O)C1 C(=O)(C1=NOC(C)C1)NCC(COC)NC(C1CCCN1N=O)=O CC1(C)CCC=C1C(=O)N1CC2CCCC2(NC(C2CCS(=O)(=O)CC2)=O)C1 N1(C(CCC2(C)CC2)=O)CCCC1Cn1cc(C2CC=CCC2)nn1 CCC(CC(=O)NC(C)CCCNC(c1cc(C(C)C)n(C)n1)=O)OC Cc1cncc(C(=O)N(C(C)CCNC(C2CC2c2cccnc2)=O)C)c1Cl N1(C(CCC)=O)CCCC1C(=O)N(C)CCOCCCNC(C1CC=CCO1)=O C(CCN=C(NCC1(C#N)CC1)NCc1ccco1)OC.C1C(=O)N1 C1(NC(CSC)=O)CC12CCC(NC(=O)CC1(C)CCCO1)CC2 CS(=O)C1(CNC(c2coc(C(=O)CNC(=O)CCOC3CCCC3)c2)=O)CC1 C(=O)(C(C#N)C(C)(C)C)N1CC(CC(=O)N(CC(C)(C)O)C2CC2)OCC1 Cc1ccc(C(=O)NCC2(C)CCN(C(=O)C3=CCCC3C)CC2)c2c1CCC2 c1(C2N(C(=O)NCCN3CC(C)(C)C3=O)CCC2)cc(Cl)c(F)cc1F CC1CN(C(c2cc(CF)on2)=O)CCCN1C(c1ccc(Cn2cccn2)o1)=O CN(C)S(=O)(=O)N(C)CC(=O)NC1CCCC(NC(c2cn(C)nc2O)=O)C1 C#CCC(C)(CC)C(=O)NCCC1CCC(NC(c2ccc(F)c(F)c2)=O)CC1 CC1C(NC(c2cc(C3CC3)no2)=O)CCN1C(=O)C(c1ccccc1)=O N1(C(C(=O)N(CC(=O)OC)C(C)C)=O)CCC(C(=O)OC(C)(C)C)C(O)C1 c1(OC)nc(C)cc(C)c1CNCCCC(=O)Nc1ccc(C)c(C)c1 C=CCC(CNC(=O)COCC(F)F)C(=O)NCC1(O)CSC1 c1(C(N2CCC3CN(C(=O)C=C(Cl)Cl)C3C2)=O)cc2c(C3CC3)cccc2[nH]1 N1(C(=O)NC2(C(=O)OCC)CC2)CCOc2cc(Cl)ccc2C1 N1(C(Cc2c(C)occ2)=O)CCN(C(c2ccc(C#N)cc2)=O)C(C)C1C Cc1cc(CNC(C2(CNC(=O)CNC(N)=O)CC(C)(C)C2)=O)cnc1C c1(NC2(C)CC(NC(CC3=CCN(C)CC3)=O)C2)nc(Cl)nc2c1ncn2C CC1(NC(C2(NC(=O)CNc3ncccn3)CCC2)=O)CC(F)C1 N1(C(C2CCN(C(C3(COC)CCOC3)=O)C2)=O)CCCC2(CCC2)C1 C(CC(O)C(=O)NCC(O)CN(C(=O)C(C)(C)C1CCOCC1)C)SC CC(C#N)NC(=O)NCCN(CC1CCC1)CC1CC1 C(CCC(C)CC(=O)N1CC2CN(c3ncc(C)c(C)n3)CC12)=C(C)C C1(NC(c2ccc(C)c(Br)c2)=O)CN(C(C2(O)CCC2)=O)CC2(CC2)C1 C12(C(N(C3CCN(C(c4ccsn4)=O)C3)CCO)=O)CCC(F)(CC1)C2 CC1=C(C(=O)NC2CC3(C2)CC(C(=O)NC2CCSC2C)C3)COCC1 C(=O)(C(C(C)NC(c1csc(Cl)c1)=O)C(C)C)NCc1ncc(CC)o1 C1(C(F)(F)F)CC(=O)N1.C(=O)(C(C(C)C)SC)NCC1CC(CCNC(C)=O)C1 N1(C(CCN(C)CC)=O)CCC(OCCCNC(c2ccccn2)=O)CC1 C(=O)(C1=CC2(CCOC2)C1)N1C(C(=O)NCC(C)C2CCC2)(C(C)C)CCC1 N1(C(C2(CC)COC2)=O)CC2(C(=O)NC3CC(C)(C(N)=O)C3)CC1CO2 c1(C(=O)NC2CCC(NC(=O)Cc3cc(Br)ccc3O)C2)cccc2occc12 C(=O)(N=c1nnn(C)[nH]1)N(C)CC1(c2cccc(Cl)c2)CCCC1 c1(C(C)C)nocc1C(=O)NCCCC1CCCN1C(c1cc(C(F)F)no1)=O Cc1ncsc1C=CC(=O)NC1CC2C(NC(=O)COc3ccon3)C2C1 C1(C(=O)NCCCC(C)NC(c2nc(CCCC)sc2)=O)SC2C=CC1CC2 Cc1[nH]cc(C(=O)NC23CCCC2N(C(=O)C=C2CCC2)CC3)c(=O)c1Cl n1(CC)cc(C(=O)NCC(c2ccc(F)cc2)NC(=O)C(C#N)C2CC2)c(C)n1 c1(C(N2CC(CCC)C(NC(c3ccc(C)s3)=O)C2)=O)c(C)cc(C)nc1C C1(C(=O)NC(CC)(CC)CCNC(=O)CN(C)CCO)CCn2ncnc2C1 CC(C)(C)CCCC(=O)NC1CC2CCC1CC2NC(=O)CCn1cc(Cl)cn1 N1(C(C2NC(=O)OCC2)=O)CC2CC1CN(C(=O)CCn1cc(Cl)cn1)C2 c1(OCC(=O)NC2CCC(N(C(=O)CCC3CCCC3)C)C2)ccc(Cl)nc1 c1(N2CCC(NC(C(C)SCC)=O)C(CO)CC2)nc2cc(Br)cnc2s1 C1(NC(C=CCOCCOC)=O)CCN(C(c2cncc(OC)c2)=O)CC1O c1(OC)ccc(CCC(C)C(=O)N2CC(NC(C3CCCC3)=O)C(O)C2)cc1 c1(NC(c2ccco2)COC)ccc(S(=O)(=O)NC2CS(=O)(=O)C2)cc1C#N c1(OCC(=O)NC23CC(CNC(C4(C)C=CCC4)=O)(C2)C3)c(F)cccc1F Cc1cc(C(=O)NCC=CCNC(C23CCCC2CC3)=O)cnc1C(F)F CC1C(NC(=O)C=Cc2cc[nH]n2)C(C)CCN1C(=O)Cn1cc(F)ccc1=O c1(C(CC)O)nc(-c2cc(-c3ccccc3)oc2C)n(-c2nc[nH]n2)n1 CCCCCCCC(F)C(=O)NCC12CCCC1CN(C(=O)C=CC(C)CC)C2 C(=O)(CCCCC(F)(F)F)N1C(CNC(=O)C=Cc2ccccn2)CC1 C(=O)(CC(C)CC(C)(C)C)NCC1OCCN(C(C(c2ccc(CC)s2)=O)=O)C1 c1(C(=O)NC(CNC(c2c(C)cccn2)=O)C(C)C)nc2ccccn2n1 CCCC(C(=O)NCCOC1CCN(C(c2ccnc(C)c2)=O)C1)C(C)C Cc1cc(C(=O)N(CC(=O)NC(C)C(C)(C)O)C)ncn1 C(C(C)(C)C(=O)NCC1(CO)CC1(C)C)N(C(=O)CC1CCCNC1=O)C c1(C(N2CCC(OC)(CNC(C3CC(O)C3)=O)C2)=O)nc2ncccn2n1 N1(C(C(CCC)NC(N)=O)=O)CCC(NC(=O)Cc2cncc(C)c2)C(C)C1 S(=O)(=O)(c1cccnc1NC(c1nccnc1C)C)NCC(C(F)(F)F)OC c1(C(N2CC(C)CN(C(C(=O)NC)=O)CC2C)=O)ccc2c(c1)CCCCN2 C1(C(=O)NC(C2CN(C(=O)C(N3CCCC(C)C3)=O)C2)C)(CSC)CC(F)(F)C1 C1(OC)CN(C(=O)CC(c2ccccc2)n2ccnn2)CC1NC(=O)CCSC Cc1ccc2c(c1)CCN(C(=S)NCc1ccc(N(C)C)cc1)C2C c1(-c2cc(C)nc(C)c2)cnc2ccc(C(=O)Nc3ccc(O)cc3Br)cn12 C1(C)(CNC(C2(C(=O)OC)C(=C)CC2)=O)CCN(C(c2ccno2)=O)CC1 CCC(CC)C(C(=O)NCC1(NC(c2cnns2)=O)CCCC1)N1CCCCC1 CN1CC2(CC2)CC1C(=O)NC(C(=O)NCC1(C(C)(C)O)CC1)C1CCCO1 N1(C(CSc2c(OC)cccc2)=O)CCC(C2CC2)C1CNC(=O)CC(C)C C(CCC)(C(=O)NC1CCCCC1NC(=O)C=Cc1cc[nH]n1)=CCC CN1C(=O)CN(CC(=O)NCCC2CCN(C(C3CC4CCC3C4)=O)CC2)C1=O S(=O)(=O)(c1ccc(Cl)cc1)NC(C)C(=O)NC1CC(C)(CNC(=O)CN(C)C)C1 CC1CC(NC(=O)CSc2ccccc2Cl)CN1C(c1ccncc1Cl)=O N1(C(c2nc(C)[nH]n2)=O)CCCC(C2CC2NC(C2(C(N)=O)CC2)=O)C1 CCCC(CC)CCC(=O)N1CCC(NC(C2(c3ccnc(Cl)c3)CC2)=O)C1C Cc1nn2c(c1C(N1CCN(C(C3CCCC(=O)N3C)=O)CC1)=O)CCCC2 c1(C(N(C(C)CCNC(C23CCC2CC3)=O)C)=O)cccc(C(F)F)c1 Cc1cccc(CC(=O)NCc2cc(C(N3CC(N4CC(O)C4)C3)=O)n(C)n2)c1 c1(C(F)(F)F)nc2c(c(=NC3COC4(CCCC4)C3)[nH]1)CCCCCC2 c1(C(C)(C)C)ccc(C(=O)NCCN2CC(C(C)(C)F)C2)cc1 N1(C(C(COC)C)=O)CC(O)CC1C(=O)NC(CO)C1(O)CC1 N1(C(c2c(C(C)(F)F)n[nH]c2)=O)CC23CCCC2(C1)CN(C(C1CC12CC2)=O)C3 c1(CCC)n[nH]c(=NCCCNC(c2ccc(OC(F)F)cn2)=O)s1 c1(CC)ccc(NC(c2cc(CC)on2)c2nnnn2CCCOC)c(OC)c1 N1(C(C2(C#N)CC(C)C2)=O)CCC(C(F)(F)F)C(NC(c2ccncc2)=O)C1 C1(CC)(NC(c2cc(C)ccn2)=O)CCN(C(=O)C(C(C)C)C2CCC2)CC1 N1(C(c2cn(CCC)nn2)=O)CC2C(C(=O)NOCCOC)C2C1 c1(C(N(C2CCN(C(=O)CC(C)CF)CC2)CCOC)=O)ncccc1Cl c1(C(N2CCC(CCNC(c3ccon3)=O)C2)=O)nsc2ccccc12 N1(C(C(C)=C(C)C)=O)CC2C(CNC(C3(C)CCC(C)C3)=O)C2C1 CC(CC(F)F)C(=O)N(C1CC1)CC1CCCN1C(=O)CC1CCCC1 N1(C(C(N)=O)=O)CC2(CCC(NCc3cc(Cl)cc(Cl)c3O)CC2)C1 c1(CC)cccc(C(=O)NC2CN(C(=O)C(C3CCOCC3)F)CC2F)c1C CCC(C#N)C(=O)N1CCC(C(=O)NCc2nc(C)c(C)[nH]2)(CO)C1 c1(CC(N2CCC(C(N(CC(CC)O)CC)=O)C2)=O)c(C)nc2ncnn2c1C c1(N(CCC)CCNC(c2cc(C)c(F)c(C)c2)=O)nc(C(C)C)nc(C)c1Br c1(C(=O)NCC2CN(C(c3ncn(CC)n3)=O)C2)ccc2nnc(C)c(C)c2c1 C1(CC)CN(C(=O)COC2CC2)CCC1NC(c1ccncn1)=O N1(C(C=COCC)=O)CCN(C(=O)C(Cc2ccccc2)NC(C)=O)C(CC)C1 C1(C(=O)NCC(C2CCC2)NC(=O)CC(F)F)CCN(c2ccc(F)cc2)C1=O C1(NC(c2n(CC)ccc2)=O)CCC(C)N(C(c2nc(C3CC3)no2)C)C1 Cc1nccn1CC(N1CCCC1C(C)NC(C1(C(N)=O)CC1)=O)=O Cc1ccc(F)cc1C1(C(=O)NCC2CCN2C(=O)CP(C)(C)=O)CC1 C(CCC(CO)NC(C1(C)CC(C)=NO1)=O)NC(CCOCCOC(C)(C)C)=O C1(C)(CNC(C=C(COC)C)=O)COCCN(C(=O)C2=NOC(C(C)(C)C)C2)C1 C1(NC(CC2ON=C(C)C2)=O)CC2CC(C1)CN(C(=O)C1CCc3snnc31)C2 Cc1cccc([N+](=O)[O-])c1C(=O)NCC12CC1CN(C(c1cn(C)nc1Cl)=O)C2 C1(NC(C=C(C)C(F)F)=O)CC2CN(C(C3CCCCC3(C)C)=O)CC2C1 c1(C(N2CC(O)(CCNC(C(C)SCC)=O)C2)=O)ccc2c(O)nnc(O)c2c1 c1(C(N(C2CCCC2)CCNC(c2c(C)cc(C)o2)=O)=O)ccc2sncc2c1 Cc1c(Br)ccc(F)c1C(=O)NC1CC1CNC(c1cccc(C(N)=O)c1)=O CCCC(C)(O)C(=O)N1CCOC(CN(C)C(c2ccc(OC(F)F)cn2)=O)C1 CCC(CC)(C(=O)NC1CC(N(C)C(c2cncc(Cl)c2)=O)C1)c1ccccc1 C1(NCC(CC=C)C)CCOC(CC)C1 N1(C(=O)NC(c2ccccc2)C)CCC(NC(c2cn[nH]c2)=O)C1 c1(NC2CN(C(c3nc(CC)sc3)=O)CC2(C)C)ccc(C(=O)OC)cc1[N+](=O)[O-] CCCCC(O)CC(=O)N1CCC(CNC(c2cc(Cl)ccc2C)=O)CC1C N1(C(C(C(C)C)NC(=O)OC)=O)CCCN(C(c2ccc(=O)n(C)n2)=O)CC1 c1(C(=O)NC(CCCNC(C2(CCCC)CCC2)=O)(C)C)c(Cl)sc(C)c1C N1(C(c2cc(SCC)ncc2)=O)C2CCC1C(C)C(NC(c1ncc(Cl)s1)=O)C2 C1(S(C)(=O)=O)(C(=O)NC2CC(C(C)NC(C3(C)CCCS3)=O)C2)CCC1 c1(CNC(CCc2cn(C)nc2)=O)cc(C(=O)Nc2ccccn2)n(C)n1 C1(CC(=O)NCC2C(NC(CCN(C)CC)=O)C2)CSc2ccccc2O1 c1(CC(C)NC(c2c(C)nsc2N)=O)ccc(Cl)cc1Cl C(=O)(CC(CC)CC(C)C)NC(C(N1C(C(CC)O)CCC1)=O)C O=C(C1=CNC2=NCCCC2=C1)NCC1(F)CC(CNC(c2sccc2F)=O)C1 C1(C(CC)=CC)CCCN(C(C2CC23CCOC3)C(=O)Nc2ccc(F)cc2)C1 C1(C#N)(OC)CC(C(=O)NC2(CNC(c3snc(Cl)c3Cl)=O)CC2)C1 C(=O)(CC(C=C)CCC)NC(C(=O)NC(C#C)C(C)C)(C)CO C1(C(=O)NC(CO)CCF)(CNC(c2cc[nH]n2)=O)CC12CCC2 S(=O)(=O)(c1cccc(Br)c1[N+](=O)[O-])N1CCC(C(=O)NCc2cnccn2)CC1 c1(COCCC(=O)NC2(C)CN(C(CCC=C)=O)C2)ccc(C(=O)CF)cc1 N1(C(CCCCOC)=O)CCC(NC(C2(N=[N+]=[N-])CC2)=O)C(CO)C1 c1(C(N2CCC(NC(=O)Nc3cccc(C)c3)C(F)C2)=O)c(C)cc(O)cc1C N1(C(C(CCCC)F)=O)CC2(CCC2)CC1C(=O)N(C)CCN(C)C1CC1 C12(NC(C3C(C)CCC3)=O)COC(C1)C(NC(c1ccc(C3CCC3)cc1)=O)C2 CC1CN(C(C2CN(S(=O)(=O)C(F)F)C2)=O)CC(C)N(C(=O)CNC=O)C1 N1(C(CC(CC)SC)=O)CCC2(CC1)CN(C(=O)CC1(C)CCC1)C2C(C)C CC(=O)C(C)CC(C)C(=O)NC(CC1CC1)C(=O)NC1CC(Cl)(Cl)C1 C1(C(=O)NC2C(NC(=O)CCOC3CCC3)C2)C2CCC(F)(F)C12 Cc1ccc2c(c1)C(CC(=O)NC1CN(C(=O)C=CCF)CCC1(C)C)C(=O)N2 c1(C(=O)NC(CC)CN(C(c2ccc(O)nc2)=O)CC)cnc2ccnn2c1N N1(C(CCC)=O)CCCC2(NC(=O)C=Cc3ncc(C)[nH]3)CC2C1 c1(SCC)cc(C)ccc1C(=O)N(CCCOCCNC(=O)C(C(C)C)OC)C N1(CC2(CCOC)CC2)CCC(=O)N(CC2(C)CCC2)C1=O c1(C(=O)NC(C2N(C(COC)=O)CCC2)(C)C)cnc(NC2CC2)c(Cl)c1 CCCC(C(=O)N1CCC2CC12C(=O)NC(c1ccccn1)CO)NC(C)=O N1(C(CSCCC)=O)CCC2(CC1)CCN(C(=O)CCF)CC2 Cc1cccc(CCNC(C2CC(O)(Cn3cc(-c4cccs4)nn3)C2)=O)c1 Cc1cc(O)ncc1C(N1CCC(C(C)(C)C(=O)NCC2(CO)CCCO2)C1)=O CC(CC(=O)NC1(CO)CCCN(C(c2cc3occc3[nH]2)=O)C1)CC(C)(C)C c1(C(CNC(C(C)NC(CN(CC)CC)=O)=O)O)cnn(C)c1 C1CS(=O)(=O)Cc2cn(nn2)CCCO1.c1(C(C(=O)NC2CC2)O)ccccn1 Cc1cc(C)c(C=CC(=O)N(C2CCC(NC(c3cccs3)=O)CC2)C)cc1C C=CC(C)(O)CC(=O)N1CCCC(C(C)C(=O)N(CCC(N)=O)CC)C1 C(c1cccnc1)=CCNC(C(C)N(C(C(C1CC1)OC)=O)C)=O C1(C(N2CC(O)(C(C)NC(C3SCCCS3)=O)C2)=O)Cc2nn(C)cc2C(=O)N1 c1(SC)cccc(C(N2CC(C)(NC(C3CCOCC3C)=O)C2)=O)c1[N+](=O)[O-] C1(C(=O)NC(CC#C)(C)C(=O)N(CC(C)CC)CC)CC(=O)CC12CCC2 c1(C(N(CC(CC)NC(c2cc(C(F)(F)F)on2)=O)C)=O)cncn(C)c1=O CC1(CNC(=O)C(F)C2CCC2)CN(C(C2CC(=O)C23CCC3)=O)CCO1 C(CCSC)(C(=O)NC(c1cnccc1C)C)NC(Cc1cn(CC)nn1)=O C1(C(C(=O)NC(C)C)N(C(CCCCC)C)C2CCCOC2)CC2(C1)OCCO2 C1(C)(C(=O)NC(C2CN(C(C3CSCCS3)=O)C2)C)COC(=O)OC1 CC1CC(C(=O)N(C2CN(C(c3cc(CO)on3)=O)C2)C)CCS1 C1(F)(C(=O)NCC2(CCNC(c3ncc(OC)cn3)=O)CC2)CCS(=O)(=O)C1 c1(COC(C)C)cn(CCC(=O)NC(c2cnn[nH]2)C)nn1 C1(CNC(Cn2cc(CNC(C3C(C)=CCS3)=O)nn2)=O)CC[Si](C)(C)C1 CCCCC(CNC(=O)CCC(=O)NCCC)NC(c1c(C)noc1CC)=O C1(C(N2CCCC2c2ccn(C)n2)=O)(CC)CCOC1 CCCCS(=O)(=O)CC(=O)NCCN(C(=O)CCOCC)CCOC(C)(C)C(F)(F)F C12(C(=O)NCC(N(C)O)=O)CCN(C(=O)CCC3(C)N=N3)CCC1C2 Cc1nc(CCC(=O)NC2CC(CCNC(c3nnn(C)c3C)=O)C2)oc1C N1(C(c2c(OC)scc2)=O)CC2C(NC(=O)CC(C)c3cnn(C)c3)C2C1 Cc1nc(C)c(C(=O)NC2CN(C(C3CCCS3)=O)CC2C(F)F)s1 Cn1cc(C(=O)NCCN2CCN(C(C3(C#N)CCC3)=O)CC2)c(Cl)n1 Cc1nn(C)c(O)c1CNC1CCC(Cn2cc(CN3CCC(O)CC3)nn2)C1 CCCC(CCO)NC(=O)C(C1CCN(C(c2ccnn2CCC)=O)CC1)C C(C1CCN(C(=O)CN=[N+]=[N-])CC1)=CC(=O)NCc1n(CC)cnn1 c1(C(=O)NCC2C(OC)C(OC)CN2C(=O)CCC2CC2)cc([N+](=O)[O-])cn1C c1(N2CCC(N(C)C(c3ncsc3Br)=O)C2)ncc2cc(Br)cnc2n1 C12(C(=O)NCCSC(C)C)CC(C)(CN1C(C1COCCC1C)=O)C2 C(C(C(C)C(C)C)NC(=O)Cn1ccc(C(F)F)n1)NC(c1c(C)oc(Cl)n1)=O c1(C(N2C(CNC(CC=C(C)C)=O)CCCCC2)=O)ccc2c(c1)CCCO2 C1(CNC(c2nc(COC)[nH]n2)=O)CN(C(C2(C)CCOC2C)=O)CC1C(F)F c1(NC(C#CCNC(C2(C=C)CCCC2)=O)=O)ccc2nc[nH]c2c1 N1(C(CN2CCC(C)CC2)=O)CC2CCCCC2(NC(C2CCCCCC2)=O)C1 N1(CC(N2C(C)(CC(=O)N(CC(C)C)CCN(C)C)CC2)=O)CCC(CO)CC1 CC(=O)n1cc(CN2CCSCC2C(=O)NOCC2CC2)c2cccnc12 N1(C(CC2CC(OC)C2(C)C)=O)CCC(Nc2ncnc(O)c2Br)C(C)C1 CCN=c1[nH]cc(C(N2CCC(N(C(=O)CCSCC(C)C)C)C2)=O)s1 C(CCCCNC(=O)CC1CCC1(C)C)NC(CCN(CCC(C)(C)C)C)=O c1(CN(CC=C)C(=O)NC2CCN(c3ccncn3)CC2)ccc([N+](=O)[O-])cc1 C(=O)(C1CCCc2c[nH]nc21)N1C2(CNC(C(CCCC)N(C)C)=O)CC(C1)C2 c1(C(c2n(CCOCC)nnn2)NCCC2C=CCC2)ncc(Cl)cc1Cl C1(C(=O)NC2CCCC2NC(=O)C(=CC2CCCC2)C)(COC)CC=CC1 c1(C(=O)NC(C(C)NC(c2cc(C(N)=O)[nH]n2)=O)CO)cc(N)ccc1Cl c1(C(C)C)ncc(C(C(=O)NC2CCN(CC(C)O)CC2)N(C)CCSC)cn1 CC(C(=O)NC12CCC(CNC(c3c(F)cncc3Br)=O)(C1)OC2)S(N)(=O)=O C1(C)(CNC(C(C)NC(CC)=O)=O)CCCN1C(c1cc(OC)ccn1)=O N1(C(CCCOc2c(C)nn(C)c2C)=O)CC2(C1)CN(C(C1CC1Cl)=O)CCO2 C1(C(N(C2CN(C(C(c3cn(CC)nc3)=O)=O)C2)C)=O)C(O)C(=O)N(C)C1C C1(C(C)NC(C=CC(C)C)=O)CN(C(c2ccnn2CC#N)=O)CCO1 C1(C(N2C(CCC=C)CCC2)=O)CC1C1CN(C(c2cccc(CO)c2)=O)C1 CCC(CNC(C1COC(=O)N1C)=O)(CC)C(=O)NCC1(OC)CN(C)C1 C(=O)(CC(=O)NC(CNC(c1c[nH]nc1C(F)(F)F)=O)CO)N(C)C c1(OC)ccc(C(=O)NC2CC(Nc3ccn4ncc(I)c4n3)C2)cc1[N+](=O)[O-] C(C1=CCC2CC1C2(C)C)(c1nnnn1C1CCCCC1)NC(CCOC)COC C1(C2CN(C(c3cccc(=O)o3)=O)C2)(NC(c2c(C)n(C)nc2)=O)CC1 CC(C)C(C)(C)C(=O)N1CCC(NC(C2OCCCC2(C)C)=O)C(F)C1 c1(CC)[nH]nc(Cl)c1C(N1CCC(CF)(NC(c2cc(C#N)c[nH]2)=O)C1)=O C(C)(C(=O)NCCN(C)CCF)(C1CCC1)NC(C(C)OCC#C)=O C1(C(=O)NCC(C)(C)NC(=O)CCCOC(C)(C)C)CCC(F)(F)C1 S(=O)(=O)(c1ccc(CC#N)cc1)N(c1ccc(F)c(Cl)c1)CC n1(CC(=O)NC(C(C)NC(C(CC(C)C)N(C)C)=O)CO)cnc2ccccc12 C1(NC(c2cccc(OC)c2F)=O)CCN(C(C2C3COCC23)=O)CC12CCC2 C1(C2CC2)(NC(c2cccc(C)c2Cl)=O)CCN(C(=O)CCOCC2CC2)C1 C1(C(=O)NC2CCC(C(=O)NCC3(CCCO)CC3)C2)CCCCCC1 C(=O)(C1=CS(=O)(=O)CCC1)N1C(C2(NC(c3c(C)cno3)=O)CC2)CCC1 c1(C(N2CCC(Nc3nc(C)nc4c3scc4)C2)=O)cc([N+](=O)[O-])c(C)cc1C c1(CNC(C2(F)CN(c3ncc(OC)cn3)C2)=O)c(OC)cccc1Br C(CC(C(=O)O)N(C(C)(C)C)C(C)=O)NC(=O)CC1(n2ccnc2)CC1 CC1=C(C(=O)N2CC(C3CN(C(c4cnc5scc(C)n45)=O)C3)C2)CCCC1 c1(C(N2C(CNC(C3(OC)CS(=O)(=O)C3)=O)CCC2)=O)cccn2cnnc12 c1(C(N2C(CO)CC(NC(C(C)CC3CCC3)=O)C2)=O)cnc2[nH]cnc2c1 N1(C(C2N(CCC)CCC2)=O)CCOC(C)(CNC(C2(CC3CC3)CCC2)=O)C1 CCCCCCC(=O)N1CC(F)CC1CNC(C1(C)CC2(CCC2)C1)=O c1(SC(C(=O)NCCC2CC(NC(c3c(C)nns3)=O)C2)C)ccc(Cl)cc1 CCC(C)CCC(=O)NC1COCCN(C(=O)C(c2cccc(Cl)c2)(C)C)C1 Cc1nc(C(C)C)nc(O)c1C(N1CCOCC(NC(C2(C)CCCC2)=O)C1)=O c1(OCC(=O)NCCC2CCN(C(=O)C3=CCC3)C2)cccc(F)c1F C#CC1CN(C(=O)CC(C)NC(=O)C(C)CC(=O)OCC)CCN1C C1(n2cc(NCC3CCC(NC(C(CC)OC)=O)C3)nn2)CCCCNC1=O C1(C(N2CCCC2C2CCOC2)=O)CC2CC2N1C(=O)C=CC1CCOC1 Cc1cc(NCC(C)(C)NC(=O)C=Cc2scnc2C)ccc1[N+](=O)[O-] c1(C(N2CC(CNC(CC(=C=C)C)=O)C2)=O)ccc(OCCC)c(C(F)F)c1 N1(C(CN(C)C2CC2)=O)CCCC(CO)(NC(=O)CCc2cc(Cl)cs2)C1 C1(NC(=O)CN2CC3CC3C2)C=CCN(C(=O)CSC2CC2)C1 O=S(=O)(c1cnc(NCCC2CCCO2)c(Cl)c1)N1CCc2ccc(Br)cc2C1 c1(C(N2CC3C(NC(c4cccc(C)n4)=O)C3C2)=O)c(C)cc(O)nc1C Cc1ccc(C(N2CCC(CCNC(c3cc(C4CCC4)no3)=O)C2)=O)cc1 C1(CC)C(C(=O)OC)CCN1C(=O)C(C)NC(=O)Cn1cnnn1 C1(NC(C(C)N(C(=O)C(C)=C(C)C)CC)=O)CCOC(C(N)=O)C1 c1(OC)cc([N+](=O)[O-])c(CN2CCC(O)C2C(N2CCOCC2CO)=O)cc1Cl Cc1cccnc1Cn1cc(CNC(=O)C(C)(C)NC)nn1 CCC(CCC(=O)NCC1CC(O)C(F)C1)NC(=O)C1CC1 C1(NC(c2n(C)ncc2)=O)CN(C(c2ccc(F)c(C(F)F)c2)=O)C2(CCC2)C1 c1(C(N2C(CNC(C(CCC)NC(C)=O)=O)CCC2)=O)c(OC)ccc(F)c1N C1(C(=O)NCc2ccc(O)cc2)Cc2ccccc2CN1C(c1ccc(Cl)[nH]1)=O c1(NC(N(C(C)Cc2ccsc2)C)=O)cccc(-c2ccnn2C)c1 N1(C(C2(CCCC)CCC2)=O)CC2(CCCN(C(C3CC(=O)N(C)C3)=O)C2)C1 n1(CC)nc(C)c(C(N2CCC(C)(NC(=O)CC3CC(CF)C3)C2)=O)c1Cl C1(NC(C(c2ccc(F)cc2)OC)=O)CC2CC1N(C(c1csc(Cl)c1)=O)C2 N1(C(C2CC(=O)NC2)=O)CCC(C2CCCCN2C(=O)CCC(N)=O)CC1 N1(C(C(CCSC)NC=O)=O)CCCN(C(C2(CF)CC2)=O)CC1C c1(C(=O)NCC(C)(C(C)C)NC(C(CC)CC)=O)cc2c(s1)CCCC2 c1(C(=O)NCC(CNC(c2ccc(CC3CCC3)cc2)=O)F)ccnnc1S CC1(NC(=O)CC2CCC(O)C2)CCN(C(c2n[nH]c(=N)s2)=O)CC1 C(C(CNC(=O)COCC1CCC1)C(F)(F)F)NC(c1cccc(C)c1)=O c1(CC)cccc(C(N2CC3C(NC(=O)C=Cc4nnn(C)n4)C3C2)=O)c1O c1(OC)ccc(C(N2CC(CNC(=O)CSC(C)C)CC2C)=O)c(C)n1 N1(C(=O)CC23CCC(CC2)C3)CCC2CN(C(c3cc(O)cs3)=O)CC2CC1 CCCCS(=O)(=O)N1CCCCC1C(=O)N(CC)CC1(C)CCCC1C C(=O)(C(Cn1cccn1)NC(C1CCCN1C)=O)N(C)CC1CC(F)(F)C1 C1(c2onc(C3CCCN(C)C3)n2)CC2(CC(NC(C3CCCN3C=O)=O)C2)C1 N1(C(C2N(C(C(C=C)OC)=O)C(C)C2)=O)CCC(OC)CC1 CCCCCC(C)CC(=O)N1CC(C2CC2)(C(N2CCOC(C)(C)C2)=O)C1 N1(C(C2C(C(N)=O)COC2)=O)CCC2(CC1)CCN(C(=O)CCc1cocn1)C2 Cc1nncc(C(=O)NCC(C)(C)CC(=O)N(C2CCCC(C)(C)C2)C)c1C N1(C(C2CC23CCSCC3)=O)CCC2C(C1)CN2C(c1cnn[nH]1)=O C(c1ccc(Cl)s1)=CC(=O)NCCCC1N(C(C=CCOC)=O)CCC1 N1(C(CCN(CC(=O)C(CN(C(C)=O)CCCC2CC2)=O)C)=O)CSCC1N.CO.O N1(C(CCOC)=O)CC2CCN(C(C3CCCC34CCOCC4)=O)CCC2C1 C1(C(=O)NC2C(OC)C(O)C2)CN(C(=O)C(n2nccc2C)C)C2(CCC2)C1 C=CC(CC)C(=O)N1CC2C(C(N3CCC(CC(C)(C)C)C3)=O)C2C1 C(=O)(C1=CCC(NC(=O)C(C(C)CC)OC)C1)NCc1nc(CC)oc1 C(C)(C)(C(C)CC(=O)NCC(O)C(=O)NC)NC(COC1(C#C)COC1)=O C(=O)(C(CN=[N+]=[N-])NC(c1cn(C)c(=O)n1C)=O)N(C)CC1CCCCO1 c1(CCC(C)=O)cn(CCCCNC(=O)C(C)(F)F)nn1 O=C1CN(C(C2CC(NC(C3(O)CCSC3)=O)C2)=O)CC(=O)N1 C(=O)(CCCC1CCCC1)NCCN(C(=O)Cn1nccc1C)CC N1(C(C(C)SC)=O)CC2CC(NC(=O)C(C(C)C)C3CCC3)C2C1 C(=O)(CC(C)(C)N(C(=O)CC1COC(=O)C1)C)N1CC(N(C)C2CC2)C1 CN1C(=O)CC(NCc2ncnc(O)c2Br)C1c1cccnc1 c1(C(=O)NCC2N(C(C(C)n3cccn3)=O)CC2)ccc2[nH]nc(Cl)c2c1 C(=O)(C(C1CCCC1)NC(=O)C=CCOCCOC)NCC(=C)C CC1(C)COCCC1CC(N1CCC1CNC(=O)C(c1ccc(Cl)cc1)CO)=O CC#CCC(C(=O)NCc1n[nH]cc1CC)NC(c1cc(OC)no1)=O Cc1cc([N+](=O)[O-])cc(C(=O)NCC(C2CCC2)NC(c2cnc(S)[nH]2)=O)n1 c1(C(=O)NCCC(CNC(C(CCC)N(C)C)=O)O)c(O)cc(Cl)cc1F C1(C2(O)CCC2)(C(=O)NCCC2(C)CCN(C(C3CCS(=O)(=O)CC3)=O)C2)CC1 c1(C(C(=O)NCC(CNC(C(C)OCC(C)C)=O)C)O)ccccn1 c1(C(C(=O)N(C2CCN(C(Cc3cc(C)sc3)=O)C2)C)=O)ccc(O)cc1 n1(CC(=O)NC23CCC2CN(C(c2ccnc(O)c2)=O)C3)nnc2c1CCCC2 N1(c2sc(C#N)c(Cl)n2)CC2CCN(C(C3CCS(=O)(=O)C3)=O)CCC2C1 C1(C(C)C)(C(=O)NCC2CC=CCC2)CCN(C(=O)Cc2cncs2)C1 N1(C(C)=O)CCC(C(C)C(=O)NCC(C)NCc2cn(C)nn2)CC1.C(CO)S C1(O)(C(C)NC(=O)CCc2cccnc2)CCN(C(=O)C(F)(F)C(F)F)CC1 N1(C(CP(C)(C)=O)=O)CCC2(CCCN(C(=O)CCCCc3cnc[nH]3)C2)C1 c1(NC)cncc(C(N2CCC(NC(c3ccoc3Br)=O)C2C(C)(C)C)=O)c1 CCC(C)C(=O)NCCC(Cc1ccccc1)NC(C1COC(=O)O1)=O c1(C(N2CCOC(COC)C2)C(=O)NCCC)ccccc1NC(=O)N(C)C c1(C(=O)NCC(CNC(c2ccc(C(C)=O)nn2)=O)(C)C)cc(Cl)cc(C)c1C c1(COC)nc(NCC2CCOCC2)cc(=NCC2CC(F)(F)CO2)[nH]1 CC#CCCCCNC(=O)C(CC=CC)NC(=O)CCC1CCCO1 Cc1nc(S)sc1CC(N1CC(NC(C2(O)CC(F)(F)C2)=O)C(C)C1)=O c1(C(=O)NCCCC(F)F)ccc2c(c1)CCOC2 C(CCCC(=O)N1CCC1(C)CC(=O)NC(c1ncccc1F)C)OCC N1(C(C(F)=C(C)C)=O)CC2(CCC2)CCC1CNC(=O)C=Cc1ncc[nH]1 c1(CNC(CN(C(C2C(CC)CCO2)=O)CC)=O)cn(C)nc1C CCC1=C(C(=O)N2CC(NC(c3cncnc3C)=O)C3(CCC3)C2)CCCO1 N1(C(CN(CCC)C)=O)CC(CNC(c2cc3c(s2)CCCC3)=O)CC12CCC2 c1(OCC)cncc(C(=O)NC2(CNC(=O)Cc3ccsc3C)CCOC2)c1 C1(NC(c2c(C)coc2)=O)CC2CCC1CN2C(c1cnn(C2CCC2)c1)=O n1(CC)cc(Cl)c(C(N2CCC2CNC(=O)C(c2ccccc2)N(C)C)=O)n1 c1(CCC)ccc(N)c(C(=O)NCC2CC(C)(C)CN2C(C2CCOC2)=O)c1 Cc1nn(C)c(C)c1C(N1CCN(C(C2(C)CC3(CC3)C2)=O)CC1)=O C1(C(=O)NC2(CCNC(C(C)C(F)F)=O)CC2)CCc2cn(C)nc2C1 C(C(=O)N(C1(C(=O)NC(C2CC2)C2CC2)CC1)C)(C1CCOC1)OC c1(C(C(=O)NC(CC)C)N(C2CCN(C)C2)C)ccc(OC)c(C)c1C Cc1ccc(C(C(=O)NCCCF)N(C(C)CC(C)C)C)cc1C#N c1(OC)ccc(C(=O)NC(CNC(=O)CC(C)C(F)(F)F)CO)c2cnccc12 N1(C(c2n(CCOC)ncc2)=O)CC(O)CC1C(N1CCN(CCO)CC1)=O N1(C(c2ccncc2)=O)CCCC(S(=O)(=O)N2CCc3sccc3C2)C1 C1(NC(C2(OC)CCSC2)=O)CN(C(=O)CCC(=O)N(C)C(C)C)CC2(CC2)C1 C1(C(N(C)CC2CN(C(c3ccco3)=O)CCO2)=O)CCCC2CCCN12 N1(C(C(C)(C)OC)=O)CCC(C)N(C(C2CCN(C)S2(=O)=O)=O)CC1 c1(C(=O)NC2C=CC(C(=O)NCCc3cc[nH]n3)C2)cc2c(cc1Br)OCO2 N1(N(CC=O)C)CC(O)C(O)C1CNC(=O)C1=C(Cl)CC1.c1(C=O)ccoc1 c1(C(N2CCN(CCCNC(=O)C(F)(F)C3CC3)CC2)=O)csc2nnsc12 C1(NC(CCOC(C)C)=O)CCN(C(=O)CC2CCCS2(=O)=O)CC1C C1(CC)CN(C(=O)Cc2ccc(Cl)cn2)CC1NC(C1CCCOC1)=O Cc1nc(-c2ccn(C)n2)sc1CC(=O)NC1CCCN(C(=O)C(F)(F)CO)C1 N1(C(=O)NCC(c2cccnc2)CC2CCOC2)CCn2c(Br)cnc2C1 c1(CSCC(=O)N(CC(C)CNC(=O)CSC2CCCCO2)C)ccc(F)cc1 C(C1(O)CCCc2ccccc21)NCCC1CCC(OC)CC1 C1(O)(CC)CCN(C(=O)C(C2CC=CCC2)NC(=O)CCNC(=O)CO)CC1 C1(OC)(CNC(=O)CC2CCCCN2C)CCN(C(c2nc(C)n(C)n2)=O)C1 C1(c2cccc(OCC(F)(F)F)c2)(NCc2ncc(C)s2)CCOCC1 C1(NC(C2(c3cc(Br)ccn3)CC2)=O)COCCN(Cc2ccnc(O)c2)C1 N1(C(CCN=[N+]=[N-])=O)CC2CCCC1C2.C1(C(=O)NC(C)(C)C)CC2CCCC12 Cc1ncc(C(=O)N(C2CCCN(C(=O)C(C)(C)C3CC3)C2)CCF)c(C)n1 CCCC(C(=O)NC1(C)CCN(C(=O)C(C(C)C)c2cccnc2)C1)N(C)C Cc1ccc(F)c(CC(=O)NC2(C)CCN(C(c3cc(N)c(Cl)cn3)=O)C2)c1 c1(C(=O)NCC2CC(C)(C)CN2C(=O)COC(F)F)ccnc2ncccc12 c1(OC)ccc(NC(C2CCCN2C(c2cnc(Br)c(F)c2)=O)=O)c(I)c1 c1(C(=O)NCC2C=CC(NC(C3(CC(C)=O)CC3)=O)C2)nc2nc(C)ccn2n1 C1(OCCN(C(=O)C(=O)OC2CC2(F)F)C)COCC1OC C1(NC(CC(=O)N(C)C)=O)CC(CC2CC2)N(C(=O)C=CSc2ccccc2)C1 c1(OC)cc(C(=O)NCCC(C)CCNC(c2ccnc(CO)c2)=O)cc(C)n1 C#CC(C)(C)C(=O)N1CCN(C(CNC(C2CC2C)=O)C(F)F)CC1 n1(CC#C)cccc1C(=O)NC1CC1NC(c1cnc(C2CC2)s1)=O C1CC(C)(C)CNC(=O)C2CCC(C(C)C)N12.c1(C=O)ccc(C(C)=O)o1.CO C1(C(=O)NCC(CN(C(c2c(OC)n[nH]c2)=O)C)O)C2CC(=O)CC12 C1(C2OCCN(C3=C4N3C4=O)C2)CCOc2ccccc2C1.CCCCCCCC Cc1c[nH]cc1C(=O)N(CCC(C)NC(c1cnn(CC2CCC2)c1)=O)C C(=O)(N=c1cc[nH]c(C)c1Cl)c1c(OC)ccc(S(C)(=O)=O)c1 N1(C(c2c[nH]c(=NC)o2)=O)CCC2(CC2C(=O)NC(C)(C)C(C)(C)O)C1 c1(C(c2nnnn2C(C2COC2)C2CC2)NCCOC)ccccc1 Cc1nc2nccc(N3CCN(C(c4ccccc4Cl)=O)C4(CCC4)C3)n2n1 C(CCC1CC1)(C(=O)N(C(C)CSC)C)NC(C(CC)n1cncn1)=O c1(CN2CCC3(C(NC(c4ccc(F)nc4)=O)C3)CC2)c[nH]c2ncc(Br)cc12 N1(C(COCCC#C)=O)CC(NC(C2CCN2C)=O)CC12CCCC2 Cc1n[nH]c(C)c1C(=O)NC1CCCN(Cc2cncc(OCC(F)(F)F)c2)C1 C(=O)(CCCN=c1nccc[nH]1)OCC(c1c(C)c(Cc2ccccc2)[nH]n1)=O CN1CCN(CC(=O)NC2CC(F)CN(C(c3ccc(CO)cn3)=O)C2)CC1=O C1(OC)(OC)CC(C(=O)NCCCOCCNC(=O)C(C)(C)SC(C)C)C1 c1(CC)ccc(OCC(O)CNC(=O)Cn2nnc(=O)[nH]2)cc1 N1(C(C(C2(O)CCC2)NC(c2scc(C)c2)=O)=O)CC2(CCC2)CC1C c1(OC)ncc(C(N2CCC(C)(CNC(=O)C3=CCOC3)C2)=O)cc1Br C1(CNC(C(CCOC)C)=O)CC2(CC2)CN1C(=O)Cc1occc1C c1(NCCC(=O)N(CCC)Cc2ccccc2)c(F)cc([N+](=O)[O-])cc1F CN1CCN(C(C2CC3(CC3)CN2C(=O)Cc2ccccc2O)=O)C(CO)C1 C1(Nc2cc(OCC)ncn2)CCCN(C(=O)CCc2ccc(Cl)s2)CC1 N1(C(CC=CCC)=O)CC2CC1CC2CNC(C1CCCCN1C(C)=O)=O N1(C(c2c(C)coc2C)=O)CCC2(CC1)CC2C(=O)NC(c1ccc(Cl)cc1)C c1(N(CC(C)(C)OC)C)nccc(=NCC(C)CN2CCOCC2)[nH]1 N1(C(c2c(OC)ccc(C)n2)=O)CCC2(CCN(C(=O)CC3(C)CC3(Cl)Cl)C2)C1 c1(C(=O)NC(C)C)ccc2c(c1)CCN2C.C12CC3CCC1CC3C(=O)N2 C12(C(=O)NC(CC)(C)CNC(c3ccn(C(C)(C)C)c3)=O)CCCCC1C2(F)F N1(C(CCC2(C)CCC(=O)N2)=O)CC2CCC1C2NC(=O)CC1(N2CCCC2)CC1 C1(NC(COC(C)(C)C)=O)C=CC(C(=O)Nc2csc(Cl)c2)C1 c1(C(N2CCC(CF)C2)C(=O)NCC)cccc(OCC(F)(F)F)c1 C(CCCC(=O)N1CCC(N(C(=O)Cn2nccc2C)C)C1)NC(C)=O N1(C(C(C)SC)=O)CC2C3CCC(C2C1)N(C(C1CC2(C1)CC(F)(F)C2)=O)C3 c1(CNC(C)CC2CC2)cccc(Br)c1Br C(C(=O)N1CC2CC1CN2C(=O)OC(C)(C)C)(C(C)C)c1cccc(C)c1 c1(NC2(CO)CN(C(Cc3cn(CC(C)C)nc3)=O)C2)cc(O)nc(O)n1 C=CC1OCCC1N=c1nc(N2CCN(C)C(C(F)(F)F)C2)c2c([nH]1)CCOC2 C(CC(O)C(=O)NC1CC(N(C(=O)CSc2nnnn2C)C)C1)N(C)C C1(C(N2CCC(N3CC=CC3)C2)C(=O)NC)CCC(SC)CC1 CC(=NO)C1CC(C(=O)NCC(=C2CN(C(c3c(C)nsc3N)=O)C2)F)C1(C)C CC1CN(C(c2cnoc2)=O)CCC1N(C(=O)Cc1cc[nH]n1)C c1(CNC(=O)NCc2ccc(N3CCCC3)nc2)cccc(-c2ccccc2)n1 n1(CCC(=O)N(C2CC(NC(C(CC)(C)CO)=O)C2)C)cnc2sccc2c1=O N1(C(C=C(C)c2cnn(C)c2)=O)C2CCC1CN(C(=O)CN1CCSCC1)C2 c1(NC2CCCC(CNC(C3C(C#C)C3)=O)C2)sc(C)c(C)c1C=O.C(=O)OC Cc1cc(I)ccc1C(N1CCN(C(c2sc(Br)nc2C)=O)C(C(F)(F)F)C1)=O N1(C(c2cc(C)c(C)s2)=O)CC2=C(C1)CN(C(=O)CC(O)Cc1ccccc1)C2 c1(OCCC(=O)NC(c2cn(C(C)(C)C)nn2)CO)cc(F)ccc1F CC1(C)CCCN(C(C2CCCS2)=O)C1C(=O)NCc1cnn(C2CC2)c1 C1(C(N2C(CCNC(=O)CC=C(Cl)Cl)CSCC2)=O)CCc2nnc(O)n2C1 c1(CNC(c2c(C)ccs2)=O)cc(C(=O)NCC(C)OCCO)ccn1 C1(C2CCCO2)(C(c2nnnn2C2CCC2)NC2(C(=O)OC)CC2)CCCC1 N1(C(c2cncc(OC)n2)=O)CC2(CCCC2NC(C2CC(N=[N+]=[N-])C2)=O)C1 CCC(C(=O)N1CCC(NC(c2cnc(Cl)s2)=O)C1)C1CCOCC1 c1(C(=O)NC2CC(CNC(c3n(C)ncc3)=O)C2)cncc2nc[nH]c12 C1(OC)CN(C(=O)CSc2cccc(C)c2)CC1NC(C12CC(CF)(CO1)C2)=O S(=O)(=O)(c1ccc(Br)cn1)N1CC(CNc2nc(OC)c(C)cn2)OCC1 C(=O)(C1=CCC1)N(C(C)CCNC(=O)C(C)SC(F)(F)F)C CN1CCn2nc(C(N3CC(C4CCN(C(=O)C5CC5)CC4)C3)=O)cc2S1(=O)=O c1(C(=O)NC2CC2CNC(c2ccsc2C(F)F)=O)cc2ccc(Cl)cc2[nH]1 CCC(O)C(C)C(=O)N1CCC(C(C)NC(C2CCN2CC)=O)CC1 c1(OC)ccc2c(N3CC(O)(c4cscc4Br)C3)nc(Cl)nc2c1 C(CCCCC(=O)NCc1cc(C(N)=O)no1)NC(C1(CC)CCCCC1)=O c1(CN(C(=NC)NCCC2CCOCC2C)C)cc(Cl)cc(Cl)c1 c1(NC(c2cnnn2C)=O)ccc(C(C)NC(C2(CN)CCC2)=O)cc1 C(=O)(CC(C)C(F)(F)C(F)(F)F)NCC(C)N(C(c1c(COC)nn(C)c1)=O)C C1(NC(c2ncc(C)c(C)c2)=O)CN(C(c2cocn2)=O)CC12CCCC2 c1(C(=O)NC2C3CN(C(C(C=C)O)=O)CC32)ccc(S(=O)CC#N)cc1 Cn1nccc(-c2ccc(C(C)(C)O)cc2)c1=O c1(OCC)c(C(=O)NCC2(OC)CCN(C(C3(C)CC3)=O)CC2)cccc1F c1(C(CC)C(=O)NCC(C)N(C)C(c2ccn(CCOC)n2)=O)ccc(Cl)cc1 CC1CN(C(=O)CC2CNC(=O)O2)CCC1CNC(C1CC2(CC2)C1)=O n1(CCC(=O)NCC2C(NC(C3(C)CCNC3=O)=O)C2)ccc2ccccc12 C1(OC)CC(CNC(=O)C(n2cc(C)cn2)C)N(C(c2cccc(O)n2)=O)C1 N1(C(c2cnc(OCC)c(Cl)c2)=O)C2CCC1C(F)C(NC(=O)C(F)C(C)C)C2 CCC(C)(C)C(=O)C(=O)N1CCC(CC(=O)NC2CCOC(C)(C)C2)C1(C)C C1(NC(C2CCC(CC)O2)=O)CCCN(C(c2ccc(C(=O)NC)nc2)=O)C1 c1(CC(=O)N(C)Cc2c[nH]nc2C(F)(F)F)ccc([N+](=O)[O-])cc1Cl N1(C(C(CC)Cl)=O)CCC2C1CCN2C(c1n[nH]c(C)c1F)=O c1(C(N2CCC(C)(CCNC(C(C)OCCCC)=O)C2)=O)ccnc2c1CCC2 C(C)(c1cccc(Cl)c1)=CC(=O)N(CC(C)NC(=O)C(O)C(F)F)CC c1(C2CCCC2NCCC(=O)Nc2ccc(F)cc2)ccc(Cl)cc1 N1(C(CSCC#C)=O)C2CCC1C(CNC(=O)C(Br)=C(C)C)C2 C1(N(C(C=CC=CCC)=O)C)CCN(C(=O)CSc2nccn2C)CC12CC2 CC1CC(C(=O)NCC(F)(F)CC2CC2)N1C(=O)CN1CCNC1=O N1(C(CN2CC(=O)NC2=O)=O)CC2CC(C1)C2NC(=O)CC12CCCC1C2 C1(C(=O)NC(C2CCCN2C(=O)CSCC(N)=O)C)CCOC(C)(C)C1 CC(C)CCC(O)C(=O)NCCC(C)NC(c1ccc(CNC(N)=O)cc1)=O N1(C(COCC=C)=O)CCC2CN(C(=O)Cc3ccc(C)c(F)c3F)CCC2C1 C=C1CC2CCC(C1)N2CC(c1ccc(OC)c(F)c1)O C1(C(N2CCC(CC#C)(C(=O)NCC3CC(C)(O)C3)C2)=O)C2CC3C(C2=O)C13 Cc1cc(C(=O)NCCOCCNC(C23CC(CO)(C2)C3)=O)nc(C)c1 c1(OC)c(CN2CCC(N(C)C(c3csc(C(F)(F)F)n3)=O)C2)cc(Cl)cc1Cl c1(CC(N2CC(N(C)C(c3sc(F)cc3Cl)=O)C2)=O)ccc(C(C)(C)C)cc1 C(c1ccc(-c2ccccn2)s1)=CC(=O)NC1CC(O)CN1 N1(c2nc(OC)c(F)cn2)C2CCC1CC(NC(C1(C)COC1)=O)C2 c1(NC(C2N(Cc3cnc(N(C)C)c(Br)c3)CCC2)=O)ccc2c(c1)CCCC2 N1(C(CCN(CCC)C)=O)CCC(CNC(c2cnn(CC(F)F)c2)=O)C12CC2 CCC(CN(C)C)CC(=O)NCc1nc(C(C)(C)C)nn1C C1(CNC(C(C)n2cncn2)=O)CCC2CN(C(c3cc(N)cc(F)c3)=O)CC12 C1(O)(CCNC(C(C=CC)O)=O)CCN(C(C2(C(C)(C)O)CCC2)=O)C1 C1(CNC(C(C)n2cccc2)=O)CCC(C(=O)NCc2ncc(CO)o2)O1 C(=O)(CCCN(C)N=O)NC1CCC(NC(C=C(C)Cl)=O)C1 C=C(CNC(=O)C(c1ccnn1C)NC(=O)C(C)CCCOC)c1ccccc1 CCCCC(C)(F)C(=O)NCC1(NC(c2n[nH]c(C)c2C)=O)CCOC1 C1(O)(NC(C(=C)F)=O)CCN(C(=O)COc2ccc(C)cc2)C1 c1(C(=O)NCC2N(C(COc3cn(C)nc3)=O)CCOC2)cnc2[nH]cnc2c1 N1(C(C2CCC(CNC(Cc3nc(C)sc3)=O)O2)=O)CCOCC(O)C1 Cc1ccc(CC(=O)NCC2CC2NC(=O)Cc2cccc(Cl)c2)cc1 N1(C2CN(C(=O)C(CO)c3ccccc3)C2)CCN(C(C2(F)CCOC2)=O)CC1 N1(C(c2ccc(C)nc2)=O)CCCC(O)(CNC(=O)C(C)c2cncs2)CC1 c1(C(C)=O)ncc(C(=O)NCC2OCCC2C(=O)NCCCCC2CC2C)s1 N1(C(CCCC#CC)=O)CCOC2(C1)CN(C(=O)C(C)Sc1ncccn1)C2 c1(C(N(CC(=O)OCC)C)=O)ccc(Br)c(Cl)c1F c1(C(N2C(CC3N(C(=O)OCC)CCC3)CCCC2)=O)cccc2c1OCC2 C1(NC(c2c(C)oc(CNS(C)(=O)=O)c2)=O)CN(C(=O)C(C)CO)CC12CCC2 c1(C(=O)NC2C=CC(CNC(c3csc(O)n3)=O)C2)cc(F)cc2nccnc12 C1(NC(C2(C(=O)NC)CCC2)=O)CC2CCC1N2C(C1CCN(C)C1=O)=O c1(ONC(C2(SC)CN(C(=O)CC=C(C)C)C2)=O)ccccc1F N1(C(CNC=O)=O)CC2CCN(C(c3ccc(-c4ccco4)o3)=O)CC12 c1(C(N(CCC)CCNC(=O)C(C)(C)n2cccn2)=O)ccc2cccnc2n1 C12CC3CCC1N3C2.Cc1ncoc1CNC(=O)C1CC1 c1(CC)cccc2[nH]c(C(N3CCN(C(=O)Cc4ccc(C)s4)C4CC34)=O)cc12 Cc1cc(=O)c(C(N2CCCCC2C(C)NC(=O)C=C(Cl)Cl)=O)cn1C1CC1 c1(C(N2CCC(CC)(NC(=O)COCC(C)C)CC2)=O)cn2nccc2nc1C C1(C(N(C2CCC2)C(C)C)=O)CC(C)N1C(=O)CCCN(C)C c1(C(=O)NC(CCNC(CCSc2nc(C)[nH]n2)=O)C)sc(C#N)cc1Cl N1(C(CC(C)C)=O)CC(CCNC(c2c(Cl)nsc2Cl)=O)OC(C)C1 C1(CC)CN(C(=O)Cn2nccc2C)CCC1NC(c1occc1Br)=O N1(C(C2CC(=O)OC2)=O)CCC(CF)(NC(=O)CCN2CCCS2(=O)=O)C1 CN1CC(C(=O)NC2(C)CCN(C(c3ccc(F)s3)=O)C2)OCCC1=O c1(CSC)cc(C)c(C(=O)NC2CN(C(c3cnc(NC4CC4)s3)=O)CC2C)o1 C1(NC(C(C(C)C)NC=O)=O)CCN(C(=O)CC2(C)CCS(=O)(=O)N2)C(C)C1 Cc1nc(NC2CCCCN(C(=O)C3CCc4c[nH]nc43)C2)ncc1[N+](=O)[O-] Cn1nnc(C(=O)NC(C)(C)CNC(C2CC(C)(C)C2)=O)c1C(F)(F)F CCCCC(CNC(=O)COCCOC)NC(=O)C=CC1CC1.c1ccccc1 n1(C(C)C)ncc(C(=O)NCCOC2CN(C(C3COC(=O)N3)=O)C2)c1Cl C(c1cnc2ccccc2c1)=CC(N1CC(C)OCC1)=O c1(C(N(CCCNC(=O)CCC(C)N(C)C)CC)=O)cnc2n1C(C)CCC2 C1(NC(c2c(C)noc2)=O)Cc2ccccc2N(C(C2CN3CCN2CC3C)=O)C1 C12(C(=O)NC(c3[nH]nc(C(C)C)n3)C)COCC1CN(C(c1cnns1)=O)C2 C(=O)(CC(F)(F)C(F)F)N1CCC(CCOC)(NC(c2c(CCC)occ2)=O)C1 c1(OC)cc(NC(C2CC(NC(c3ccnn3C)=O)C2)=O)cc(OC)n1 c1(CCC)ncc(C(=O)NC2CCN(Cc3nc(CC4CCCC4)no3)C2)s1 Cn1cc2cccc(C(N3CCC(NC(c4n[nH]cc4F)=O)C(O)C3)=O)c2n1 CCC(C)C(O)C(C)C(=O)NCC1(O)CN(C(C2(CO)COC2)=O)C1 c1(C(N2CCC(CN(C(CNC(CC)=O)=O)C)C2)=O)cnc(O)cc1O CC#CCCCC(=O)NCC(C1CCN(C(c2ccc(N)cc2C)=O)CC1)(C)O C1(CC(=O)NC(CCOC)CNC(=O)CCc2csc(C)n2)CCCC12CC2 c1(C(C(N2CC(COC)(CNC(=O)CC(C)NC(N)=O)C2)=O)C)c(C)n[nH]c1C c1(C(=O)NCC2C3CN(C(=O)C=CCn4cncn4)C2C3)[nH]cc2c1CCCC2 c1(OC)cccc(O)c1OCC(=O)NCCCCC(C)NC(=O)CC1C=CCC1 C(C(C)CS(C)(=O)=O)NC1(SCCC)CCOCC1 C1(C2NCC(CC(=O)OCC)C2)CC=C(C)CC1 c1(N2CC(CC(C)NC(c3cnn(C)n3)=O)C2)nc2ccc(F)cc2s1 c1(C(=O)NCC2CN(C(C(C)N3CCC3)=O)C(C)C2)ccc2oc(O)nc2c1 c1(C(=O)NC2CN(C(c3cc(C)on3)=O)CC2O)cc(S(C)(=O)=O)ccc1F C(C)(C(=O)N1CCCC1)N(CC)CC.C1(C)CN1.C1CN1 Cn1cccc1C=C(F)C(N1CC2C(CNC(=O)CC3CC=CCC3)C2C1)=O c1(CC(=O)N(CCCOCc2cccnc2)CCN2CCNCC2)sc(O)nc1O C1(CNC(c2nc(C)c(C)s2)=O)CC2(CCN(C(C3(C)CS(=O)(=O)C3)=O)CC2)C1 C1(NC(CC=C=C)=O)CC2(C1)CC(C(=O)NCC(C)C(C)C)C2 N1(C2CN(C(c3cc(COC)on3)=O)C2)CCN(C(C2CCCC(=O)N2)=O)CC1 CC(C(C)(C)C(=O)N1CCCC(C(N)=O)C1)NC(c1ncccc1Cl)=O N(C1CCCc2c[nH]nc21)C(CSCCNC(Cn1ccc(C)n1)=O)=O c1(C(=O)NC2C(C(N3CCC(N(C(C)=O)C)C3)=O)C2)nc(C)c(C)[nH]c1=O C1(NC(CNC(C(CC)(F)F)(C)C)=O)CCCC1S(C)(=O)=O C1(C(=O)NCCC2N(C(C(CC)CO)=O)CCSC2)CC2(C1)CC(C)(C)C2 C12(C(=O)NCC3N(C(c4cc(C)nnc4)=O)CCC3)CCC(CF)(C1)OC2 C1(C(=O)NCC2OCCN(C(c3cccc(C#N)c3)=O)C2)CN2CCCCC2CO1 c1(SCC(=O)OC(C(=O)NC2CCC(C)CC2)C)cc2ccccc2[nH]1 C1(NCC)CCCN(C(=O)C(=O)NC2CCN(C3CCNCC3)C2=O)C1 N1(C(c2c(C#N)nc[nH]2)=O)CCCC12CCN(C(c1cnc(O)o1)=O)CC2 C1(C(=O)NC2C(NC(Cc3nccc(OC)n3)=O)C2)Cc2cccnc2C1 CN1CC(O)CC1(C)C(=O)Nc1cnc(Cl)cc1C(F)(F)F CC1=C(C(=O)NCCCN(C(=O)CC(F)(F)Cl)Cc2ccccc2)SCCO1 N1(C(=O)Cc2ccc(Cl)cc2)CCN(C(c2cccnc2O)=O)C(CC2CC2)C1 C(C)(N=c1[nH]c(=NCCc2ncc(Br)cn2)[nH]c2cc[nH]c12)c1c(C)ncs1 c1(N(C)CC2CCCN(C(C(C)N3CCCC3)=O)C2)c(Cl)cccc1[N+](=O)[O-] N1(C(CS(CC)=O)=O)CC2CC(C1)C2NC(=O)C=Cc1ccc(C)cc1 c1(C(N2CCC(OCC(=O)NCC3N(CCC)CCC3)C2)=O)cc(O)ccc1C Cc1cccc(OCC(=O)NC2CCCN(C(c3cnc[nH]3)=O)C2C)c1F C1(CC(=O)N(CC(CNC(c2cc(C(=O)OC)[nH]c2)=O)(C)C)C)CC2(CCC2)C1 c1(C(C(=O)NCC2(CNC(=O)C3CC3)CC23CCC3)(F)F)ccc([N+](=O)[O-])cc1 C1(CCC(=O)NC2(CCO)CCOC2)CCN(C(C2CC3(CC3)CO2)=O)CC1 c1(CC)cc(C(N2CCCCC2Cc2cn(C3CCC3)nn2)=O)nn1C c1(C(C(=O)NCC2CC2)N(C(CC)C(=O)OC)C)cc2nc(Cl)ccc2o1 CC(C)C(O)CC(=O)NCCCNC(c1ccc(CCO)cc1)=O c1(OCC)nc(Cl)ccc1C(N1CC(CC(=O)OC)C1)=O c1(OC)cnc(Cl)[nH]c1=NCC1(NC(=O)C2=CS(=O)CCC2)CCCC1 C(C1OCCc2ccccc21)n1c(N2C(C)C(=O)NCC2)nnc1CSC1CC1 C1(C2N(C(COCC=C)=O)CCC2)CCN(C(c2ccccc2C)=O)CC1 N1(C(CC)(C)CNC(=O)NC(C2CCC(C)CC2)CO)CCc2sccc2C1 c1(C(N2CC(C(C)NC(c3cc(F)cs3)=O)OCC2)=O)cnnc2ccccc12 N1(C(C2(C#C)CC2)=O)CCC(C(=O)NCC(CC(C)C)N(C)C)C(O)C1 C1(CC(=O)NCCCC(C)NC(C=CC)=O)CN(C(C)=O)CCO1 c1(C(N2CC(CC(C)NC(C(C)N(CC)CC)=O)C2)=O)cnn2ccn(C)c12 c1(NC(=O)NCC(C)(C)NC(c2n[nH]c(C(C)(C)C)n2)C)cnn(CC(F)F)c1 CCCCN=c1[nH]c(=NC(C)Cn2cnnc2)c2c(ncn2C)[nH]1 O=C1CCCCC(C(N2CCC2C(=O)NCCn2ccc(=O)cc2)=O)N1 C1(NC(c2c(OC)nsc2OC)=O)C(C)CN(C(=O)Cc2nocc2C)CC1C c1(C(=O)NCC2N(C(c3cncc(CC)c3)=O)CC2)c(O)ccc(F)c1Br c1(C(=O)NCCOCCN(C)C(C2CCCC(=O)O2)=O)nc(=O)n(C)[nH]1 Cn1ccc(F)c1-c1cccn1C1CCN(C=O)C1.C(CC(F)(F)F)NCCO CCCC(CNC(c1cnnn1C)=O)NC(c1cscc1OC)=O C1(NC(C2(C)N(C(C3C(C)N(C)CC3)=O)CCC2)=O)CN2CCC1(C)CC2 N1(C(C(CC=C)C)=O)CCN(C(c2sc(Cl)cc2Cl)=O)C2COCC12 O=Cc1cccc(CC(N2CCC(CN3CCCCCC3CO)C2)=O)c1 C1(C(=O)NC2CCC(N(C(=O)Cc3csc(Cl)n3)C)CC2)CCn2nccc2C1 c1(OC)c(C(N2CC(N(C(=O)CN(C)C3CC3)C)C2)=O)ccc(Cl)c1Cl C1(NC(C(C)OC(C)(C)C)=O)(CNC(=O)C2=COCCO2)CCC(F)(F)CC1 Cc1nnn(CC(=O)NC(C)CNC(c2cc(C3CC3)[nH]n2)=O)n1 S(=O)(=O)(c1ccccc1F)N1CCC(N(CC)CC)C1.c12cc(c(Br)cn1)CO2 c1(CC)cc(Cl)ccc1C(N1CC2CC1CN2C(=O)C(C)C#N)=O C1(NC(CC(=O)NC)=O)CC2CCC(C1C)N2C(C1(C)CC2CCC(C1)S2)=O c1(OC)ccc2c(C(=O)NCC3C=CCN3C(=O)C(F)C(F)(F)F)cnn2c1 CCC(CC)CC(F)C(=O)NC(C1(O)CCN(C(=O)C=CCN(CC)CC)C1)C C1(NC(c2c(C)nc(C3CC3)[nH]2)=O)CC2CC1CN2C(=O)Cc1cccs1 CCC(C(=O)NCC(C)C(=O)Nc1cc(C)c(C)cc1C)C(C)(C)CC N1(C(CC2(C)CCN(C(=O)CN3C(=O)CCCC3=O)C2)=O)CCC(C2CC2)C1 N1(C(COc2cn(C)nc2)=O)CC=C(C(=O)NC2CC(C)(C)OC2=O)C1 N1(C(C2C(C)(COC)C2)=O)CCC(CO)(NC(=O)C(c2csc(C)n2)=O)CC1 C1(N(C(C(N2CCN(C)CC2)C)=O)C)CCN(C(c2cc(Br)co2)=O)CC12CC2 c1(NC(C2CC=CCC2C(N2CCC(CC3CC3)C2)=O)=O)ccc(CO)nc1 N1(C(=O)Cn2nnc(=O)[nH]2)CCC2(CCCN2C(c2csc3ccccc23)=O)C1 N1(C(CNC(=O)OCC=C)=O)CCC(CN(C(c2cn(C)nn2)=O)CC)CC1 c1(C(=O)NCCOC(C2CC(CN(C)C)C2)=O)c(F)cc(F)cc1F c1(CNC(C(CC)COC)=O)cccc2c1CN(C(=O)CCCCC(C)C)C2 C1(C(=O)NCCC(C)NC(C23CCN(CC2)C3)=O)CC2C=CC1C2 C=CCC(C)(CC=C)NC(C1C(C)CCN1C(=O)COC)=O C1(C(=O)NC(C)(CNC(=O)CSc2ccc(F)cc2)CO)CC2(CCCC2)C1 c1(C(N2CCC(CO)C2C)C(=O)NC(C(=O)OC)C)cccc(C(F)(F)F)c1C C1(NC(CN(S(CC)(=O)=O)C)=O)CCCN(C(=O)C2=NNC(C(F)(F)F)C2)C1C CC1=C(C(=O)NC(C(=O)NCC2CC2CO)c2ccoc2)CCO1 CC(C)CC(C)(O)C(=O)N(C1(CC(=O)NC2CC23CC3(F)F)CC1)C c1(CC(=O)NCC2C(C(N(CC(C)N(C(C)=O)C)C)=O)CC2)c(C)noc1C Cc1cc(Cl)c(C(=O)NC2CC(NC(=O)CCc3nccn3C)C(O)C2)cc1F N12CC(CC(C(C)(C)C)C1)NC(=O)C2=O.N1(CCCC)CCOCC1C(=O)OC c1(CC)nnc(O)c(C(=O)NCC2CCN2C(C2(C)CCCN2C)=O)c1CC c1(N(C)CC2CCCN(S(=O)(=O)c3ccncc3)C2)ncnc2ccccc12 c1(C(=O)NC(CNC(=O)C2=CCOCC2)C2CCC2)ccc2nn[nH]c2n1 Cc1cc(C(=O)NC2CCC2NC(=O)CC(C)(C)C)c(N)c(Cl)c1 C1(C(=O)NCCN(C(=O)CCCCN2C(=O)CCC2=O)CC)CC(S(C)(=O)=O)C1 S(=O)(=O)(CC(=O)NCC1C2CN(C(=O)CC3C=CCCC3)CC12)NCC c1(NC(C2(C(=O)OCC)CCCN(C(=O)NC3CC3)C2)=O)ccc(C#N)cc1I c1(OC)c(C)ccc(C(=O)N(C2CN(C(c3csc(Cl)n3)=O)C2)C)c1F C1(NC(C2C(C)=C2)=O)CC2CCC(C1)N2C(c1ocnc1-c1ccccc1)=O C1(C)(C(=O)NCCOC(C)=O)CCN1C(=O)C(O)c1ccco1 N1(C(=O)NC(C)CN(c2ccccc2)C)CCC(c2ccccc2)CC1C C1(CN(C)C)COCCC1(F)F.C12CC13CC(C3)NC(=O)c1ccc(o1)C(=O)N2 C12CCCCN1C2=O.c1(NC(C)CO)nccc(Oc2ccccc2)n1 C(C)(C(C)NC(=O)CNC(c1cscn1)=O)NC(C=C(C)Cl)=O N1(C(c2c(SCC=C)cccc2)=O)CC2(CCC2NC(=O)C2=CC(C)(CC)C2)C1 C(CC(CC)C(=O)NC(CC(F)F)C(=O)N(C)Cc1cncn1CC)=CC CCC(C)CC(=O)N(C)CC1CCN(C(=O)CCNC(C2CCCCC2)=O)CC1 N1(C(CC(=O)OC)=O)CCN(C(=O)CCCCCSC)C(CC(F)F)C1 Cc1cc(C)c(CC(N2CC3C(CNC(=O)CNC(c4cscn4)=O)C3C2)=O)s1 c1(N2CCC(C(C)NC(C3CCOC3)=O)C2)ncc([N+](=O)[O-])cc1CO N1(C(C(CC)(C)OC)=O)CC2(CCN2C(c2ccccc2CCC(F)(F)F)=O)C1 CCCC(CC)CCC(=O)N(C(CC)C(=O)N(CC(=O)OC)CC1CC1)C Cc1cc(NC(=O)CC2CCN(C(=O)CC(C(C)C)c3ccccc3)C2)cnc1F CCC(O)(C(=O)NCC(O)CNC(c1cc(OC)ncn1)=O)c1ccccc1 C1(C(=O)NC(C2(O)CCN(C(c3cscc3Cl)=O)C2)C)CCCC(C)C1 N1(C(c2c(C)nc(C(C)C)s2)=O)CCC(C)(CNC(=O)Cc2cccs2)CC1 CCC(CN=C(NCc1nc(C(F)(F)F)cs1)NC1CCS(=O)(=O)C1)C(=O)OC C1(C(=O)NCC2(CCNC(C3CCC(C)(C)O3)=O)CC2)COCC(C)(C)O1 C1(CN2C3(CC(Cn4cc(CSC)nn4)C3)CC2)CC2COCC(C1)C2 c1(OCC)ccc(C(=O)NCCCOCCNC(C2C(C)C2C)=O)cc1N N1(C(=O)NCCCC=CC)CCCOC(c2ccccc2Cl)C1 C1(NC(C2CN(C)C2)=O)CCN(C(=O)C(C)(C)c2cnco2)CCC1CO C1(NC(=O)COC2CCCCC2)CCN(C(c2ccc(I)c(O)c2)=O)CC1O Cc1nc(N2CC(C(=O)NCC34CCCC(CO3)C4)CC2C)c2ccsc2n1 N1(C(C)=O)CCN(C(=O)CCN(C(C2CCC3CC23)=O)CC2CC2)CC1 c1(C(=O)NCC(CNC(CCc2cc(C)on2)=O)F)ccc(N)c(Br)n1 Cc1cccc(C(N2CCC(C)(CNC(C3CCC(=O)C3)=O)CC2)=O)c1C c1(NC(c2cn(CCNC(C3C=CCS3)=O)nn2)=O)ccc2ncnn2c1 C1(CCC)CCC(O)(C(=O)N(C)CCn2cc(CC(C)(C)C(=O)O)nn2)CC1 C1(C(C(=O)NCC=CCNC(C2C(CCOC)C2)=O)C)CCCCCCC1 N1(C(C(C2CCN(C(c3c(C)scn3)=O)C2)F)=O)CC2CCC(C1)C2O C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CN(C(c2cc(=NC)[nH]cc2)=O)C2C1CCC2 C=CCCC(F)(F)C(=O)NC1CCCCC1NC(C1CC(=O)NC(=O)C1)=O C=CCCCCCC(=O)NCC1(CO)CCN(C(C2(F)CCN(C(C)(C)C)C2)=O)C1 Cc1nn(C)c(Cl)c1C=CC(N1CC(C)CN(C(=O)C(Cl)=CCl)C(C)C1)=O c1(C(=O)NC(C)CNC(=O)COCC2CC2)cccn2c(O)nnc12 C1(OC)(OC)COC(CNC(c2ccc(C(F)F)s2)=O)C1 CCC(C(=O)NCC1(CNC(=O)C=NOC)CCOCC1)C(C)O N1(CC(=O)OC)C(=O)NC2CC1(CN1C3CCC1C(CC(=O)OC)C3)C2 C(C)(C(C(=O)NCCc1cccnc1)C(C)C)NC(c1cccc(C)c1N)=O C12(NCC3(S(C)=O)CC3)CCC(C1)OC2 c1(C(C)NC(c2c(C3CC3)cnn2C)=O)ccc(F)cc1F c1(N2CC(F)CC(C(=O)NCc3ccc(C)c(C)n3)C2)ncnc2occc12 N1(C(=O)CC2CC23CC3)CC2(CCN(C(c3cn(C4CCCCC4)nn3)=O)C2)C1 N1(C(Cc2c(C)ccnc2)=O)CCC2(CCN(C(C3COCCC3C)=O)C2)C1 CCCCCCC(O)CCC(=O)NCC1CC(NC(C2CCCC(=O)CC2)=O)C1 C(CC(O)C(F)(F)F)NC(CCC1(NC(CCC2CC(C)C2)=O)CCC1)=O C1(NC(c2cn(C3CCCC3O)nn2)=O)CCN(C(C2CCCOCC2)=O)CC1 n1(CC(C)C)nc(-c2ccc(F)cc2)nc1C(F)(F)CC1CC1 CC1CCN(C(C2CCCN(C(c3c(F)cccc3F)=O)CC2)=O)CCO1 c1(OCC)ncc(C(=O)NCC2(NC(C3C=CCCC3)=O)CCOC2)s1 N1(C(c2c(SC)cn(C)n2)=O)CCC(NC(=O)C(F)C(F)(F)F)C12CC2 C1(CNC(C2C(C)OCC2)=O)CC2(CC(NC(c3cnn(C)c3C(F)F)=O)C2)C1 N1(c2ncc(SC)cn2)CCC(NC(c2cc(Cl)cnc2F)=O)C(F)C1 C1(CNC(C2CC(F)(F)CS2)=O)(CO)CCCN(C(C2(O)CCC2)=O)C1 c1(OC)cc(-c2ccncc2)ccc1CNCc1ncccc1OC C1(CC=C)(NC(=O)Cc2ccccc2CC)CCN(C(c2ccncc2Cl)=O)C1 C1(CNC(=O)COCCO)CC2(CC2)CN1C(C1CC2CC2C1)=O c1(CN2CC(O)(CNC(=O)Cc3cccc(C(F)F)c3)C2)[nH]nc([N+](=O)[O-])c1Cl C12(C(=O)NCC3C(NC(C(CCC)=CCC)=O)CC3)CC=CCN1CCC2 c1(CN2CCN(C(c3c(OC)c(Br)ccc3)=O)C3C2C3)ccc(C#N)cc1F N(C(=NCCOC1(C)CCCC1)NCCOC(C)C)C(CCCC)C CC(CCCCNC(c1cc(C#N)c[nH]1)=O)NC(c1cc(C(F)F)no1)=O C(=O)(CS(=O)(=O)CCO)N(C)CC1CCCN1C(=O)CCc1cnn(C)c1 c1(C(N2CCC(NC(C(C)(C)c3ccsc3)=O)C(O)C2)=O)c[nH]c2cccnc12 Cc1cccc2c(C(=O)N(C(C)CNC(C3CCc4nccn4C3)=O)C)c[nH]c12 C12(C(=O)NC3CN(C(=O)OC)C3)CC1CCN2C(c1cccc(CO)c1)=O C(=O)(C1=C2CCCN=C2NN1)N1CC(OC)C(NC(=O)C(F)CC(C)C)C1 C12(C(=O)NCCCC(C)NC(C3CC=CCC3)=O)CCCN(CC1)C2 c1(C(=O)NC2C(CN(C(C3C(C)CN(C)C3)=O)C)CCC2)ccc(N)c(F)c1 c1(OCC(=O)NCC(C2CC2)NC(C(C)NC(CC)=O)=O)ccccc1 c1(CN(C)C(N2CC(c3c(F)cccc3F)(O)C2)=O)ccc(Cl)cc1Cl c1(N(C2CCN(C(CCC(=C)Cl)=O)CC2)C)snc(Cl)c1C#N C1(NC(C(C)OCCN(C)C)=O)COCCN(C(=O)Cc2cccc(N)c2)C1 Cc1nn(C)c(Cl)c1-c1cn(C2CC(C(N3CCS(=O)CC3C)=O)C2)nn1 C(=O)(C(N=[N+]=[N-])C(C)C)NC(CC(=C)C)C(=O)NC1C=CCC1 C(=O)(CCCC(C)(C)C)NCC1C(C)CCCN1C(=O)Cc1csnn1 N1(C(CCC(=O)OCC)=O)CC(NC(C2(CCF)CC2)=O)CC2(CC2)C1 CCC(C)(C(=O)NCCC1CCN(C(=O)CC2CCN(CCF)CC2)CC1)OC c1(CNC(=O)NC2(C)C(C)CCC2)cc(F)c(Cl)c([N+](=O)[O-])c1Cl CC1(C)CN(C(c2nc(Br)cs2)=O)CCC1NC(c1ncc2ccccn12)=O Cn1cc(Br)c2c(I)cnc(NC3(c4ccc[n+]([O-])c4)CC3)c12 c1(C(C)C(=O)NCCN2CCN(C(=O)C3=CCC3)CC2)ccc(F)c(F)c1 Cc1cccc(C(=O)NC(C(=O)NC(Cc2ccco2)CO)c2ccoc2)c1N N1(C(c2ncsc2NCCCC2CC2)=O)CCCC(CCC=O)C1.CO c1(OC)cc(C)nc(N2CCCC2CNC(=O)C(n2nc(C)cc2C)C)n1 Cc1csc(C)c1C(=O)N(C)CC1CCN(Cc2ccc(C(N)=O)cc2)CC1 N#Cc1cccc(I)c1NC(C1CC(NC(c2c(F)cc(F)cc2F)=O)C1)=O c1(C(N(CC)CC2CCN(C(=O)CC(C)C)CC2)=O)cc(N)nc(Cl)c1 C(=O)(CS(=O)(=O)C1CC1)NC(CNC(C1(C#C)CCCC1)=O)C(C)C C(=O)(C(C)C1CC1)NCCCN(C(CC1(COC)CC1)=O)CCO C1(NC(C(COCC)C)=O)CCCCCC1C(=O)NC(C)C(C)(C)O N1(C(c2ccc(C)o2)=O)CC(NC(=O)CC2CCCNC2=O)C(CO)C1 c1(CC(=O)NC(CN(C)C(C2CC2(C)C)=O)(C)C)cc(F)cc(F)c1 Cc1nc(NCc2cnc(CC3CC3)s2)cc(N2CCC(CC3CC3)C2)n1 n1(CC)nc(C(=O)NCC#CCNC(=O)CCN2CCCS2(=O)=O)c(C)n1 C1(C(=O)NCCC(CC)(C)NC(=O)C(N2CCNC2=O)C)CNC(=O)CC1(C)C N(C(=NCCC(=O)N(C)C)N1CCSC(C)(C)C1)CC(CC)C(C)C Cc1cc(NC(C2(O)CN(C(=O)COc3ccccc3F)C2)=O)ccc1Br CC(C)(C(=O)NCCn1cnnn1)C1=CCN(C(=O)Cn2cccnc2=O)C1 C1(CNC(C(CC)(C)OC)=O)CC2CC1CN2C(=O)CCc1ccc(F)cc1 CCCC(C)CCCC(=O)N1CCOC(CNC(c2nccc3n[nH]cc23)=O)C1 C(=O)(CC1CCc2ccccc21)NCC1(F)CN(C(CC(CN(C)C)(C)C)=O)C1 CCC(C)(COC)C(=O)N(C1CCN(C(C2CC3C=CC2CC3)=O)CC1)C c1(NC(c2cncc(CNC(C3N(CC)CC3)=O)c2)=O)cccc([N+](=O)[O-])c1 CC(=O)C(C)CCC(=O)NCCOc1ccc(C(=O)O)c(Cl)c1 C(=O)(C(F)C(C)(C)O)N1CC=CC(C(=O)NCC(COCC)C)C1 Nc1cc(C(=O)NCC(CO)NC(C2(C3CCCCO3)CCC2)=O)cc(F)c1 C1(NC(=O)C(F)CC2CCCC2)(CNC(=O)COc2ccon2)CCCCCC1 C(=O)(C(F)C(C)(C)O)N(c1ccccc1F)CCNC(C(C)(c1ccccc1)OC)=O S(=O)(=O)(CC(=O)N(C1(C(=O)NCCC(=O)NC(C2CC2)C2CC2)CC1)C)NC Cc1c(Cl)c(C(=O)N(C2CCCC(NC(c3sccc3F)=O)C2)C)nn1C C1(CC)(CO)CN(C(=O)CC2CCN2C(c2csc(CO)n2)=O)C1 c1(OC)ccc(C(N2CCN(C(=O)CCCCF)CC2C(C)C)=O)c(C)c1 C(=O)(CC(C)P(C)(C)=O)NCCN(C(=O)CCn1ccnc1C)CCC C(=O)(C(C1=CCCSC1)N1Cc2c[nH]nc2C1)Nc1c(OC)cccc1 Cc1cc(C)n2ccc(C(N3CCN(C(=O)C(=O)C(F)(F)F)CCC3C)=O)c2n1 C(C)(CCC(=O)N1CCCCC1CNC(C1(C)CC(C)=NO1)=O)OCC C1(n2cc(C3(CC)CCC3)nn2)CCCN(C(=O)C(C)c2ccco2)CC1 CC1(C)CN(C(=O)COCP(C)(C)=O)C(CNC(=O)Cc2cncc(F)c2)CO1 c1(CCC(=O)NCC2(CNC(c3c(NCC)scn3)=O)CC2)cc(C)cc(C)c1 C1(CC(=O)NC2(C(N(C)CC3(CO)CCC3)=O)CC2(C)C)CCCCCC1 c1(C(=O)NCCCC(C)NC(c2snc(O)c2Cl)=O)ccc2c(c1)CC(=O)N2 c1(C(=O)OC)cc(=NCCCNC(C2CCCN(C(=O)CSC)C2)=O)[nH]c(C)n1 Nc1ccc(C(=O)NCC(c2ccc(O)c(O)c2)O)cc1-c1nccs1 CC1CN(C)CC(C(=O)N(C)CC2CC(F)CN2C(c2cn(C3CC3)nn2)=O)O1 C1(CCNC(C2N(CC)CC2)=O)CC(F)(F)CN1C(c1ccc(CO)cc1F)=O CC1(C)CC2C(CN1CC(O)C(F)(F)F)C2(F)F S(=O)(=O)(c1cc(Br)c(F)cc1F)N1CC(NC(C2CCCCO2)=O)C(F)C1 C1(C(N2C3C(C(=O)OC)C(C3)C2)=O)CCN(C(C2CCCCCC2)=O)CC1(C)C c1(C(C(=O)NC(CCN(C(CC(C)n2ccnc2)=O)C)(C)C)C)ccccc1F CCC(F)C(=O)N(CCCN(C(=O)C(C)OCCc1ccc(Cl)s1)C)C Cc1ncsc1CSCC(=O)NCCn1cc(CO)nn1.C1(C=O)CCCO1 c1(CC)cccc(CC)c1NS(=O)(=O)C(C(C)C)c1ccc(C)cc1.C1(C(=O)N)CC1 c1(C(=O)NC(C)CCCCNC(c2ccncc2F)=O)cc2sc(Cl)cc2[nH]1 C1(CN(C(C=COCC)=O)C)CN(C(=O)CCc2scnc2C)CCO1 C(C)(C)(C(=O)NC1CCCC1CNC(=O)CNC(=O)CN(C)C(C)=O)OC N1(C(c2c(CC)ccs2)=O)CC2CC(C(=O)N(c3ccsc3)C)CC2C1 c1(C(=O)NCC(c2ccccc2)CNC(C(OC)OC)=O)ncc(C(F)F)s1 CCCC(CC)C(=O)NCC1CN(C(c2ccnn2CCOC)=O)C(C)(C)C1 c1(C(=O)NC23CCN(C(COCC(=O)OC)=O)CC2C3)cc2ccccc2nc1C C(=O)(C(O)CCCNC(=O)C(C)(C)CO)N(CCOCCOC)C1CC1 C12(NC(c3ccnc(O)c3)=O)CCCC1N(C(=O)C=C1CCCC1)CC2 N1(C(c2cc(C(F)(F)F)cs2)=O)CCCC(N2CCN(C(C3CC3F)=O)CC2)C1 c1(CC)oc2ccccc2c1CC(=O)NC1CCCC1NC(C1(CC)CCC1)=O CC(C)C(C(=O)NCC#CC(=O)NC(C1CCCO1)C)NC=O C1(C(=O)NC2(C(=O)OC(C)(C)C)CCC2)OC2CCC1CC2 Cc1c(NC(c2csc(C(F)(F)F)c2)C)ncnc1N1CCC(C)C1 Cc1cnncc1C(=O)NC1(CO)CN(C(C2C3COCC23)=O)C1 C12(CCNC(C(C)(C)OC)=O)CCC1CN(C(=O)CC1(O)CCOCC1)C2 Cc1cc(CC(N2CCCC(C(C)NC(c3snc(Cl)c3Cl)=O)C2)=O)n(C)n1 c1(C(N2CC3C(CNC(C4C(C=C)OCC4)=O)(C3)C2)=O)ccc2c(c1)CCCN2 c1(C(=O)OC)cc(C(=O)NCC2CC(NC(c3sccc3Cl)=O)C2)cs1 c1(C(=O)NCC(CNC(=O)CN=S(C)(C)=O)OC)ccc(=O)n(C(C)(C)C)n1 CCCC(CC)C(=O)NC12CC(CNC(C3CC4C=CC3C4)=O)(C1)OC2C CCCC(C(=O)OCC)NC(=O)C1CCNC2CC(C2)C(=O)N1.N(C)(C)CC C(CCCC(=O)NC1(C2CCCN2C(C2CC2=C)=O)CC1)OCCC=C Cc1cccc2ncc(C(=O)NCC(C)(C)NC(C3CCCC(CF)C3)=O)n12 C(=O)(CCCCCN(C(=O)CCON)C)NC(c1nc(=O)o[nH]1)C CC(=O)C(C)CC(C)C(=O)N1CCC=CC1C(N1CCNC(=O)C1)=O c1(-c2cn(C(CC)C)nn2)cn(C)nc1CNC(c1n[nH]cc1I)=O C#CCCC(O)CCNC(C1COCC1NC(=O)C(O)CSC)=O c1(C(=O)NC(C(C)NC(C=CCCC)=O)CO)c[nH]nc1S(N)(=O)=O c1(C(=O)NC(CC=C)CNC(C2CC3(CCC3)CO2)=O)ccc2oc(O)nc2c1 N1(C(c2c(Cl)cc(C)s2)=O)CC(NC(C2(C)CC(O)CN2C)=O)CC2(CC2)C1 N1(C(C(c2ccccc2)C)=O)CC(C)CN(C(=O)CC2CC(C)(C)CO2)C(C)C1 N1(C(C2C(CC)N(C(=O)NC)CC2)=O)CC(N2CCOCC2)C2(CC2)C1 C(=O)(C(C)(C)C(C)C)NCc1ccc(C)cn1 c1(C(C)(C)C)csc(C(=O)NC2CCC(CNC(=O)CSC(F)(F)F)C2)c1 C1(CNC(c2cc(C)no2)=O)CCN(C(c2cc(F)ccc2Cl)=O)C12CC2 c1(C(N2C3C(NC(Cc4cc(OC)ncc4)=O)C(C3)C2)=O)c(C)ncn1OC N1(C(C2(OC)CCN(C(Cc3cc(OC)no3)=O)C2)=O)CC(=O)N(C)C(C)C1 N1(C(=O)NCC(c2ccccc2)N(C)C)CCS(=O)(=O)C2(CCCCC2)C1 N1(C(C2C=CC(NC(C=Cc3c(C)cccc3)=O)C2)=O)C2CCC1CC1(CC1)C2 Cn1ncc(Br)c1C(=O)NCCOCCCNC(C1(C)CCCCC1)=O c1(CCCC(=O)NCC(C)N(C)C(c2csc(CO)n2)=O)nc2ccccc2[nH]1 C12(CN(C)C)CC(CN1C(=O)CCNC(=O)CC1CNC(=O)O1)C2 C1(C(=O)NCC2CC2CNC(=O)C(F)(F)c2ccncc2)CCC12CCC2 N1(C(CC)=O)CCC(C(N2CCCC2CNC(=O)C(O)Cc2cnc[nH]2)=O)C1 CC(C)C(CCC(=O)NC(C)CCCC(F)(F)F)NC(=O)C(C)(C)C c1(NC(N(CCN(C)C)CCO)=O)c(C(C)(C)C)nc2n1CCCC2 Cc1cc2[nH]c(C(=O)NCC(C)CN(C)C(C3CCCC(C)CC3)=O)cc2s1 c1(C(=O)NCC2CN(C(=O)Cn3ccnn3)CCO2)cc2cc(Br)ccc2s1 CCCCC(CNC(C1(F)CC1C)=O)NC(=O)CN(C)C(C)=O c1(C(N)=O)n[nH]c(=NC2CCC3CN(C(c4ccc(F)c(CO)c4)=O)CC3C2)s1 C(=O)(C(C)(F)C(C)(C)F)N1CC(O)(C(C(=O)Nc2c(CC)cccc2F)F)C1 c1(OC)ccc(C(=O)NC2CC(NC(c3cc(=O)c(C)c[nH]3)=O)C2)c(N)c1F c1(N2CCC(C)(CC)C2)ccc(S(=O)(=O)N2CCOC(C)(C(F)F)C2)cc1C#N C(C(C)(O)C(=O)NCC1(C)CCCN1C(C1CSCC(=O)N1)=O)SC CC1=C(C(=O)N2CC=CC2C(N2C3CCC2CC3)=O)CCO1 N1(C(c2c(C)cno2)=O)CC(CNC(=O)C(C)OCCN(C)C)C(O)C1 N1(C(C(C(CC)C)O)=O)CCCC(C2(NC(=O)Cn3ccc([N+](=O)[O-])n3)CC2)C1 c1(OC)ncc(Cl)c(C(=O)NC2(C(=O)OC(C)(C)C)COC2)n1 C(=O)(CC(CC)C(C)C)NCC(C(=O)NCCCOCC#C)O c1(C(=O)NCC2C(NC(c3cc(C4CC4)no3)=O)CCC2)nc[nH]c2nccc1-2 CC1CN(C(=O)CCc2ccc[nH]2)CC1NC(c1ccc(-n2cnnn2)cc1)=O c1(OC)cc(C)c(C(N2CC3CN(C(=O)C(C)(C)O)C3C2)=O)cc1OC C1(OC)CC2CC(NC(=O)CC3CC(O)CN3C(C3CCCN3C)=O)CC12 N1(C(C(C=C)O)=O)CCC(F)(CNC(=O)C(F)(F)c2csc(Cl)c2)CC1 c1(NCC2C3CN(C(c4c(C)nc(N(C)C)s4)=O)CC32)ncc(Cl)cc1[N+](=O)[O-] N1(C(Cc2cn(CC)nc2)=O)CCC(CCOC)(NC(C2CCN(C)CC2)=O)C1 c1(C(N(CCC(=O)NCc2cncc(Cl)c2)C2CC2)=O)nccc2[nH]ccc12 CCCC(CC)C(=O)N(C(C(=O)NCC1CCN(C)CC1)C1CC1)C Cc1cc(C(=O)NCCC(C)N(C)C(c2cccc(C(=O)N(C)C)c2)=O)sc1C N1(C(C(C(CC)O)C)=O)CCc2ccccc2C(N(C)C(=O)C=CBr)C1 n1(C(C)C)cnc2c(NCc3ccc(Br)cn3)[nH]c(=NC(C)CCC3CC3)nc12 C1(NC(CCCN(C(C)C)C)=O)CCCCN(C(c2cc(C#N)cs2)=O)C1 CC1CC(O)CCN(CCC(N)=O)C1.C12CN(CCO1)C(=O)CCn1cc2nn1 S(=O)(=O)(CCc1ccccn1)NC(=O)NC(CC)COC(C)C C(CC(=O)N(CC1CC1)OC)C1CCN(C(C2C(C(=C)C)OCC2)=O)CC1 CCC1=C(C(=O)NC(C2CN(C(C3CC4CC3C3CC43)=O)C2)C)CCCO1 C1(CSC)CCC(N=c2[nH]c(N(C)Cc3c(C)cccc3C)nc(=N)[nH]2)CC1 C1(CNC(C2(CC#C)CC2)=O)(OC)CN(C(=O)C(C)OCCCOC)C1 CCC(C(=O)NCc1cc(C(N2CC(O)(C(N)=O)C2)=O)co1)n1ccnc1 CC1(C)C=C(C(=O)N2CCOC(CNC(=O)C(=Cc3c[nH]cn3)F)C2)C1 c1(C(N2CC(C)C(NC(c3cc([N+](=O)[O-])c[nH]3)=O)C2)=O)c(F)cc(F)cc1Cl C#CCCC(=O)NCC#CC(=O)N(CCN(C)C)CCOC C1(c2n(CCOC)nnn2)(NCCn2ncnn2)CCN(C)C1C c1(C(N2CC(NC(C3CCC4C3C4(F)F)=O)C2)=O)cc2cccn2c(O)n1 C1(NC(CSCCCC)=O)CC2CCC1CC2NC(=O)C=Cc1cnc(C)s1 C1(C(N2C(CSC)CCC2)=O)COCCN(C(c2cnc(C)s2)=O)C1 c1(C(=O)NCC(CN(C(C2CCN(C)C2)=O)CC)(C)C)ccc(C)cc1SC CCC(C)(C)CC(=O)N(C1CCCC1)CCNC(=O)C(CCOC)OC c1(N2CC3C(OC)(CC3)C2)nc(=NCc2nncn2C)[nH]c2c1SCC2 CCCCC(CC)NC(=O)CNCP(C)(C)=O C1(C)(CC)CCC(C(=O)NCC2C3CC2N(C(=O)CCC(N)=O)C3)O1 N1(C(c2ccc(CC)cc2)=O)CCC(CNC(=O)C(c2cccs2)SC)C(C)C1 C1(C(=O)NC2C(NC(=O)Cc3nc[nH]n3)CCC2)CC2(C1)CC(F)(F)C2 C1(CNC(=O)Cc2ccsn2)CCC12CCN(C(=O)CNC(c1ccoc1)=O)CC2 [N-]=[N+]=NC1CC2(C(N3CC(CNC(c4cc(C(F)(F)F)no4)=O)C3)=O)CC12 N1(C(c2c(C)ccnc2)=O)CC2(C1)SCCC2NC(C1CCCC(C)C1)=O N1(C(C2N(C)CC2)=O)CCOCC(C(=O)NC2CC(O)C2O)C1 N1(C(Cc2nnc(C)o2)=O)CC2(CC(CC(=O)Nc3cccc(C(C)O)c3)C2)C1 C(CCCCC(=O)N1CCC(C)(C(=O)N(C)CC2(OC)CCC2)C1)=CC C1(NC(c2cnc(C)s2)=O)C2CN(CCCOCCOC(C)C)CC12 c1(C(=O)NCCC(C)(C)NC(Cc2ccc(C)o2)=O)cc2n(n1)CC(C)(C)CO2 CN1CC2CC2(NC(=O)CC2CCN2C(=O)C(F)F)C1 c1(OCC(N2CC(NC(c3n(CC#C)ccc3)=O)C2)=O)cc(C)cc(C)c1 c1(-c2ccc(C)o2)nn(C)cc1CNC(N1CCCC1c1ccccn1)=O C1(C(N2CCC(OC)C2C)=O)CC2(CCN1C(=O)C(O)Cn1cncn1)CC2 CC1CCCCN1CCC(=O)NC1CN(C(=O)COc2ccccc2C(F)F)C1 CC(C)CC(O)CC(=O)N1CC2CC2(CNC(=O)CCC2CC2(Cl)Cl)C1 C1(NC(C(c2c(C)n[nH]c2C)C)=O)CC2CCC1N2C(=O)C=Cc1cccn1C N1(C(C(COC(C)C)(C)C)=O)CCC2C(C(N3CC(SC(F)F)C3)=O)C2C1 C1(OC)CC2(C1)CC(C(N1CCC(O)(CN(C)C(C3CNC(=O)N3C)=O)C1)=O)C2 c1(NC2(c3nnnn3C)CC(CC)N(C3CC3)C2)cc([N+](=O)[O-])cc([N+](=O)[O-])c1 N1(Cc2ccc(OC(c3ncccn3)=O)cc2)CC2CCCCCCC12 Cc1ccc(C(N2CCCCC(NC(=O)C(C)(C)c3nncn3C)C2)=O)c(C)n1 N1(C(CC2C(CC)C2)=O)CCC(C)(NC(c2ccc(Cn3cncn3)cc2)=O)C1 N1(C(c2nc(CCCC)sc2)=O)CCN(C(C2CCC2(OC)OC)=O)C(CF)C1 c1(C(=O)NC2CC(NC(C3OCC4CCCC34)=O)C2)ccnc2c1CCC2 C#CC1(C(N2CC(CN(C)C)C2)=O)CN(C(c2ccnc(C)n2)=O)C1 C1(C(=O)NC(C(=O)NCC2(CO)C(C=C)C2)CC2CCCC2)CC(C(C)C)=NO1 C1(c2cn(Cc3ccc(C)cc3)nn2)CCCCCN1C(c1[nH]ccc1C)=O c1(C(N(CC(C)NC(CN2CC(CC)C2)=O)C)=O)cncc(C)c1C N1(C(C2CN(C(c3ccc(C)nn3)=O)CC(C)C2)=O)CC2(CCC(=O)N2)C1 C1(C(N2CCN(CCNC(c3c(C)ncnc3)=O)CC2)=O)C2CC3C(C2=O)C13 C1(CCC(=O)NCC(CC)N(C(=O)Cn2ccc(C3CC3)n2)C)CNC(=O)N1 c1(C(N2C(CNC(=O)C(F)n3ccnc3)CC2)=O)cccc(C(F)F)n1 Cc1c(Br)sc(CC2(NC(=O)CC(C)n3ccnc3)CC2)c1Br C(=O)(C(CCOCCO)NC(=O)CC1(O)CCOC1)N(CC)CS(=O)(=O)CC C1(NC(C(C)CCCc2ccccc2)=O)CCCC(N=c2nnn(C)[nH]2)C1 c1(COC)cccnc1C(=O)NCC(O)CNC(c1c(C)csc1Cl)=O C1(CN(C(=O)COC(F)F)C)CN(C(C2CCS(=O)(=O)N2)=O)CCO1 C1CCCNC(=O)C2CC(C2)CNC1=O.C1CCN1C(C)(C)C.CSC CC(C)CC(C)C(=O)NC1CC2CC1N(C(c1ccn(-c3cccnc3)n1)=O)C2 N(C1CCCc2cccc(F)c21)Cc1nc(N(C)C)[nH]c(=N)n1 C(C(C)(CNC(C1CCCOCC1)c1nnnn1C1CCCC1)CO)OC CC1Cc2c[nH]nc2C(C(=O)Nc2nc(-c3cc(F)c(Cl)cc3Cl)cs2)C1 CN1CCOC(C(N2CCCC2C(=O)NC(C)(C)CCN(C)C)=O)C1 c1(Cc2nc(C(CCC)C)nn2CCN2CCOCC2)c(F)cccc1Cl N1(C(C(C(C)C)OCC)=O)CCCC(C)(NC(=O)CC(C)(C)N(C)C)C1 c1(C(=O)NCC(C)(CO)NC(c2c(C)ncn2C)=O)ccc(C)c2ccccc12 O=C(C(CC(F)F)NC(C1CC1Cl)=O)NCC1CC1 c1(C(=O)OC)coc(C(=O)N(CC(C)CNC(=O)C(c2cnn(C)c2)OC)C)c1 C(=O)(CCCCCCCC)NC(CCN(C(c1cncc(C=C)c1)=O)C)C Cc1nc(C(=O)NC(C)CN(C)C(C2C(F)(F)C23CCC3)=O)cc(O)n1 c1(CC2(NC(C3(C(=O)OCC)CC3)=O)CC2)cc(Br)cc(Br)c1 Cc1sc(=O)n(CC(=O)NC(C)(CNC(C2CC(F)(F)C2)=O)C2CCC2)c1C C1(C(N2CC(CNC(c3nocc3Br)=O)C2)=O)CCCCC1C1CC1 N1(C(COCCC=C)=O)CC(C)(C(N2CCC(CCCC)C2)=O)C1 C(=O)(C1=C(Cl)CCOC1)NC1(CNC(c2ccc(Br)cc2F)=O)CC1 N1(C(=O)OC(C)(C)C)CC2CCC1CN2C(C1CCN(C(=O)C(F)(F)Cl)C1)=O CCCC(C(=O)NC1CC(C(=O)NC(C23CCC(CO2)C3)C)C1)NC(N)=O CCC(CC)(CCNC(=O)CC1COCCO1)NC(c1csc(C(C)C)n1)=O CC(C(=O)NCC1CN(C(c2cnsn2)=O)CCCO1)S(N)(=O)=O c1(C(N2CCN(C(=O)C=Cc3ccoc3)C(CF)C2)=O)cc2n(n1)CCCC2O N1(Cc2cc(C)c(Br)s2)CCC(F)(F)CC(C)C1 C1(C(N2CC3C(NC(c4cccc(C)c4Cl)=O)C3C2)=O)CC(=O)NC2CCCCC12 C1(C(C)NC(=O)C(=O)Nc2nc(-c3cccs3)cs2)CCCOC1(C)C Cc1ccc(-c2ocnc2C(=O)NC2CCC2CNC(C2CC3(CC3)C2)=O)cc1 C1(C)(CNC(C(C)C)=O)CCCN(C(c2ccncc2-c2ccccc2)=O)C1 c1(NC(C2CC3CCC2N3C(=O)Cc2ccccc2I)=O)cc(CO)ccc1F C1(C(N(CCN(C(C)C)C(c2ncnc(O)c2F)=O)C)=O)CC12CCCCC2 CCC(C)(CNC(=O)CN(C)C(C)C)C(=O)NCC(CO)N(C)C c1(OC)ccc(C(=O)NC2CCC2NC(=O)C(C(C)C)N(C)C)c(N)c1Br c1(C(=O)NCC(CCCC)NC(C2CC(F)(F)C2)=O)ccc2nccc(C)c2c1 c1(C(=O)NC(CC)CNC(C2(C)CCC(=O)N2)=O)cc([N+](=O)[O-])nn1C C1(C(=O)O)CCN(Cc2cccc(-c3ccco3)c2)CC1F CC(C(=O)NCc1coc(C2CC2)n1)S(C)(=O)=O N1(C(CC(=O)NCC)=O)CCC2CN(C(=O)C(C(C)C)SCC)CC2C1 N1(C(C(C)NC(c2ccccc2)=O)=O)CCC(C2OCC2(F)F)CC1 c1(-n2c(C3C(C)(C)NC(=O)C3)nc(CC3CC4CCC3C4)n2)cc(Cl)c(Cl)c(Cl)c1 c1(C(C)C)c[nH]nc1C(=O)N(C1CC(C(=O)NCCC2CCCOC2)C1)C C(=O)(C(C)(C)C(F)(F)F)NC1CC(C)(CNC(c2cnc(C(F)F)s2)=O)C1 Cn1ccc(S(=O)(=O)NCCC2CCN(C(c3cccnc3C(N)=O)=O)CC2)n1 c1(CC(N2CC(OC)(CNC(C3CC3C(C)(F)F)=O)C2)=O)c(C)nn(C)c1C c1(C(N2C(C(=O)NCCn3c(C)nc(C)n3)CC3CC32)=O)c[nH]c2c(Br)cccc12 N#Cc1ccc(C(N2CC(NC(c3cc(Br)nc(Br)c3)=O)C2)=O)c(F)c1F Cc1cc(C(=O)N(C(C)CN(C)C(C2CCSC2)=O)C)c2cccnc2c1C C(=O)(CCP(C)(C)=O)N(C(C)(C(N1CCOC(C)(C)C1)=O)C1CC1)C c1(C(=O)OC)c[nH]cc1C(=O)NCCCCCNC(C1(c2cc[nH]n2)CC1)=O CN1CCCC1CCC(=O)NC1CCN(Cc2cn(CCN3CCNC3=O)nn2)C1 C(C)(CCC(=O)N1C(CNC(c2cc(C(N)=O)co2)=O)CC2CC12)OC C=CCC(C)(C)CC(=O)NC1COCCC1NC(=O)CCc1cscn1 Cn1ncc(S(=O)(=O)N(CCc2ccccc2)Cc2ccccn2)c1Cl C=C(Cl)CC(C(=O)NC1CC(C(C)O)C1)NC(=O)CC(C)(F)F c1(CC(=O)NCC2CC2NC(c2[nH]cc3c2CCC3)=O)cc(O)nnc1O c1(C(N2C(C)CCC(NC(c3c(C)ncs3)=O)C2)=O)cc(F)c2[nH]nnc2c1 O=C(C1CCCn2ccnc21)NCCC1=CCN(C(c2cc(CO)on2)=O)CC1 C1(O)(CNC(C(CSCC)NC(=O)CCC2CC2(F)F)=O)CCOCC1 C(=O)(C(C(C)NC(=O)C(CO)C(F)(F)F)C(C)C)N(C1CCCC1)CC N1(C(C2C(NC(c3nc(CCC)oc3)=O)C2(C)C)=O)CCOCC(O)C1 c1(C(N2CC(c3cn(CCCCCC)nn3)OCC2)=O)cc(Cl)c(F)c(Cl)c1 c1(OC)ccc(CC(=O)NC23CC2CN(C(=O)C(F)(F)CN(C)C)C3)c(Cl)c1 c1(CC(C)C)ccc(C(=O)NNC(=O)c2sccc2Cl)cc1Cl Cc1ccc(CC2(C)CN(C(c3cnn(CC(O)CO)c3)=O)C2)o1 c1(C(N2CCC(NC(C=C(CC)C)=O)(CF)C2)=O)ccc(C)cc1Br C1(NC(C2N(CC)CCC2)=O)CCC(C)(CNC(C2(OC)CCC2)=O)CC1 N1(C(C2C(C(=O)OC)CC2)=O)CCC(F)(C(=O)NCc2nncn2C)C1 C1(C(N(CCCNC(C2CCCCO2)=O)C)=O)CCC2(CCC2)CO1 C12CCC(CC1)NS(=O)(=O)C2.C(C)(C)(C(=O)OC)OCC=C c1(C(=O)NC(C(=O)NCC(C)(CO)OC)COC(C)C)cc[nH]c(=NC)c1 N1(c2cc(OC)nc(OC)n2)CCCC(C2CC2NC(C2CC3CCC2O3)=O)C1 CCC(O)C(C)C(=O)NCC1CCN(C(=O)Cc2ccc(O)c(O)c2)C1(C)C Cc1nnccc1C(=O)NCC1CC1NC(c1ccc(C(C)(F)F)cn1)=O N1(C(CC2CN(C)C2)=O)CCSCC1CCNC(C1(C(F)(F)F)CC1)=O N1(C(CC2(OC)CCC2)=O)CCCC2(CNC(c3ccc(O)nn3)=O)CC12 C1(N(C(c2sccc2Cl)C(=O)NCCCC)C)CC(OCC)C1(C)C C1(NC(CCNC(=O)OC)=O)CCCCCN(C(=O)C=C2CCOCC2)C1 N1(C(Cc2cn(CC)nc2)=O)CC(CCNC(c2c(Cl)noc2C)=O)OC(C)C1 N1(CC(=O)NCC2N(C(C3N(CCC)CCC3)=O)CC2)CCC(O)CC1 CC12CCOC(CNC(=O)C(CCF)NC(C3C4(CC4)C34CC4)=O)(C1)C2 N1(C(C(CCSC)OC)=O)CC2(CCC2)CCC1CNC(C1CC(F)(CF)C1)=O c1(OC)ccc2[nH]cc(C3CCN(CCC(C)(C)OC)CC3)c2c1 c1(C(=O)Nc2cccc(C)c2I)[nH]nc2ncc(-c3cc4sccc4s3)cc12 C(CCCC(=O)N1CC(NC(=O)C(c2ccccc2)F)C(CC2CC2)C1)N(C)C CCCCC(C)CCC(=O)NC1(CC)CCCN(C(=O)C(=O)N=S(C)(C)=O)C1 O=C(CCS(=O)(=O)C1CCCC1)NCC1CCN(C(=O)C(F)CC2CCCC2)C1 N1(C(=O)CC2(CO)CC2)CCCC(C2CCN(c3ncc4ccsc4n3)CC2)C1 c1(C(=O)NC(CC)(C)C)ccc(CNC(=O)CC(C)SC)nc1 C1(CNC(CCC#CC)=O)C(C2CC2)CCN1C(C1CCCC1O)=O c1(C(N(C(C)Cc2cccc(C)c2)CC)=O)ccc(OC)c(C)c1 c1(C(=O)NC(C2N(C(CC(CC)(F)F)=O)CCC2)C)cc(F)c(F)c(F)c1 C1(n2cc(OCCN(C(C)=O)C(c3ccc(OC)nc3)=O)nn2)CCCC1(C)O C=CCC(C)C(=O)N1CCC(C)(CNC(=O)CC2(CS(C)(=O)=O)CC2)C1 N1(C(c2c(CC)onc2)=O)CC2(C)CC1C2NC(=O)C(C)NC(=O)COC Oc1cc(CNc2cccc(OC3CCOC3)c2)ncn1 c1(C(=O)NC2CC(CNC(C3(n4ccnn4)CC3)=O)C2)cc(F)c(Cl)cc1F CN1CCOC(C(N2CC(NC(c3ccc(C#N)o3)=O)C(n3ccnn3)C2)=O)C1 N1(C(C=C(CC)C)=O)CC(CCNC(=O)CCc2ccc(SC)cc2)OC(C)C1 Cc1sccc1C(N1CCCC1C1CCN(C(=O)C=Cc2cn[nH]c2)C1)=O c1(OCC(=O)NC(C)C(C)NC(c2cnn(C)c2Cl)=O)ccc(S(C)(=O)=O)cc1 Cc1cnn(CCCC(=O)NCC2(C(N)=O)CN(C(c3scnc3C(F)F)=O)C2)c1 C1(C(N2CCC(C)(NC(c3[nH]c(=NC)sc3)=O)C2)=O)CCc2nc(O)[nH]c2C1 C=C1CC2(C1)CC(C(=O)NC1(CN3CCN(C(=O)C=CI)CC3)CC1)C2 c1(C(CO)NC(C=CC(=O)OCC)C)cccc(C)c1 c1(C(=O)NCCCOCCOCCNC(C(C)=C(C)C)=O)c(C)cnn1C C(=O)(CC(CC)C(C)(C)C)N(CCC(=O)NCCCCC(C)C)CC#C C1(C(=O)NC(C(=O)N(C(C=C)C)C)CC2CCC2)CCCC(O)C1 N1(C(C2CCCN(C(CCCC3C(C)C3)=O)C2)=O)CC2C=CC1CC2 CCCCC1C(=O)N1C1CC1.c1(C(=O)NCC)cc(COCC)[nH]n1 CC1(C)OC2(C(N3CCCC(CNC(=O)C(F)(F)CO)C3)=O)CCC1CC2 CC1CCCC(C)N1CCC(=O)NCC1(CNC(=O)OC(C)(C)C)CC1(F)F Cc1ncc(C(N2CCCC(CO)(NC(C3CCCCN3C)=O)C2)=O)cc1C#N C1(CNC(C2(F)C(C)OCC2)=O)CCN(C(=O)CCCC(=O)C2CC2)CC1C c1(C(=O)NCC(=C2CN(C(C(c3ccc(Cl)cc3)C)=O)C2)F)ccc(CO)nc1 N1(C(C(C)CN(C)C)=O)CCCC(CC(=O)NCc2ccsn2)CC1 C(=O)(CC1=CCN(C(C2CCC2(OC)OC)=O)CC1)NC(COC)C(C)C c1(OC)c(C)cc(C(=O)NC(C)C(CO)NC(c2[nH]nnc2C2CC2)=O)cc1Cl CCCCC(C(=O)NC1CCOCC1(C)C)NC(=O)COCC(C)C C1(NC(C2CC3(CC3)CN2C(c2ccncc2)=O)=O)CCc2nn[nH]c2C1 C=C=C(C)CC(=O)NCc1ccc(C(N2CCC2C(=O)OC)=O)s1 C1(NC(C2C(=C)C2)=O)CCN(C(C2CC23CCSCC3)=O)CC1F C=CCC(F)(F)C(=O)N1CCC(F)(C(=O)N(CC(N2CCCC2)C)C)C1 CN1CCC(C(=O)NCC2(NC(=O)CCCC3CCCCO3)CCCC2)CC1 C1(N(C(C2C(CCC)C2)=O)C)CCCN(C(=O)C(F)(F)C2CCOCC2)CC1 CC1(C)CN(C(=O)CC2(C#N)CCC2)C(CNC(=O)CCF)CO1 c1(CC)cncc(C(N2CCCC(C(C)C(=O)NCCCCN3CCC3)C2)=O)c1 c1(OC)ccc(NC(C)=O)c(CN2CC(C)(CNC(c3cc(O)n(C)n3)=O)C2)c1 C=CC(C)(O)C(=O)N(CCCN(C)C(c1cc(CC)ccn1)=O)C N1(c2cc(NC(C3CC4(CCC4)C3)C)ncn2)CC2C3CCC(CC3)C2C1 c1(C2(C(=O)NCC3(C(=O)NCC4CCS(=O)(=O)C4)CC3)CC2)ccc(F)cc1Cl C(=O)(CCN1C(=O)COc2ccccc21)N1CC(NC(=O)C(F)F)C(C(F)F)C1 N1(C(C(C)n2ccnc2)=O)CC2=C(C1)CN(C(c1cc(Br)co1)=O)C2 N1(CCC(CC)C2CC2)CCN(C(=O)Cc2ccccc2)CC1 c1(C(N2C(C)CC(CC(=O)NCC3(C#C)CCC3)C2)=O)ncc(C)cc1F c1(C(=O)NC2CC2CNC(=O)C(Cc2ccccc2)C2CC2)ncccc1Cl N1(C(c2ccccn2)=O)CCN(C(c2csc(-c3ccco3)n2)=O)C2(CCC2)C1 N1(C(C(C(C)C)NC(=O)CC2CCC2)=O)CCN(C)CC(C)C1 C(C1c2ccccc2CCN1C(=O)CCCC1CC1)NC(CC#N)=O c1(C(=O)NC2CN(C(C3CN(C(C)=O)C3)=O)C2)c(C)nc(C)n1O c1(C(N(C2CCN(C(=O)C(CC)CCOC)C2)CCC)=O)nc2cccnc2s1 C=CC1(C(N2CCC(C)(N(C)C)CC2)=O)CCN(C(C2CC2C#N)=O)C1 N1(C(C(C=C)C)=O)CCC(C(CO)NC(=O)CCCn2ccnc2)CC1 N1(C(C(COC)(F)F)=O)CCc2sccc2C1CNC(=O)C(C)OCCC(C)C C(CCCC(=O)NCCCNC(=O)C(=O)C(C)C)N(C)CCO N1(C(c2cc(C#N)sc2)=O)CCCC(F)(CNC(c2ncc(F)cn2)=O)C1 c1(OC)ccc(C=CC(N2CCC(C)CC2CNC(=O)C2=C(C)OCC2)=O)nc1 c1(C(N2C(C(C)NC(=O)C=Cc3ccsc3)CCC2)=O)cnn(C)c1N C1(CCNC(C(C2CCCCC2)NC(COCC)=O)=O)CC=CCC1 C1(C(=O)NCC2CCN2CCCCC2CCC2)(COC)CCC1 C1(C(N2CCC(CNC(C3CCN(C4COC4)C3)=O)C2)=O)(OCC)CCCCC1 c1(C(=O)NCC2C(NC(c3c(C)cn(C)n3)=O)C2)cc2ccccn2c1 C(=O)(C(O)CNC(C1CCCO1)=O)N(CCC(=O)OC)CC=C C1(CC)CC(C(=O)NC(C)(C)CN(C)C(c2ccnc(OC(C)C)c2)=O)CCO1 CC1CN(C(c2sccc2S(=O)(=O)N2CCCC(C)C2)=O)CC(CO)O1 CC1CN(C(C23CC(CN2C2CC2)C3)=O)CCC1CNC(=O)CC#N C1(C(N(C(C)CN(C)C(C2(C)CCSCC2)=O)C)=O)CC2C(C1)C2(F)F C1(C(N2CCCC(C)(O)CC2)=O)C2CCC(CC2(F)F)N1C(C1CC1(F)Cl)=O C(CC(C)C(=O)NC1COCCC1C(=O)NCC(=O)N(C)O)OC c1(CC)c(Br)c(C(N2CCN(Cc3cccc(I)c3F)CC2CC#N)=O)nn1C N1(CC)CCCN(C(=O)CN(C(=O)C(N2CCOCC2)C)C2CCC2)CC1 c1(C(N2CCC(NC(c3nccc(Cl)c3F)=O)C2)=O)cnc(C2CCC2)nc1O C=CCCCCCC(=O)NCC1CN(C(=O)CSC(F)(F)F)C1 c1(C(=O)NC(C)(C)C(=O)NCC(F)CO)cccnc1O C1(NC(CCOCCCOC)=O)CC2CN(C(c3cscn3)=O)CC12 CC(O)(C(=O)NCC1CC(O)(CNC(=O)CC2CNC(=O)O2)C1)C1CCC1 C1(CCCC)CN(C(=O)CCCNC(N)=O)CCN1C(=O)COc1cnn(C)c1 Cc1nnc2n1CCCC2C(=O)NC1CCCC1NC(c1ncc(F)cc1F)=O N1(C(C2CCC(CC)O2)=O)CCC(CN(C2CCCCC2)C(=O)CC#N)C(C)C1 C1(NC(c2cn(CCC)nc2)=O)CCCCC1NC(c1ccoc1C(C)C)=O c1(C(C)=O)ccc(C(N2CCCC2CNC(C2CC3C=CC2O3)=O)=O)cc1F c1(C(=O)NCCN(C(C2(CC)CC2(F)F)=O)C2CC2)cc(OC)cc2c1OCC2 C1(C(C)NC(c2cnc(C)s2)=O)CCN(C(C2(O)CCSCC2)=O)CC1 N1(C(C(C(C)(C)C)O)=O)CCC2CC(CNC(C3(C)CC3(F)Cl)=O)CCC2C1 N1(C(c2ccc(CNC(=O)C(O)C3CCCC3)o2)=O)CCC(O)C12CCCC2 c1(CNC(C2(C)CC2(Cl)Cl)c2ccc(C(=O)O)o2)cccc2c[nH]nc12 C1(NC(C(C)(C)c2cccs2)=O)CC(O)CN(C(c2occc2F)=O)C1 C=CC(CC)C(=O)NCC(C)(CNC(=O)Cn1cnnn1)OC c1(C(=O)NC2CC(C)CN(C(=O)CSc3nncs3)C2)nccc2ncncc12 c1(C(=O)NCC2C(CNC(C(C)(C)CO)=O)C2)ccc2c(c1)C(=O)NCCO2 Cc1cccc(C(N2CCN(C(=O)CCCn3ccnn3)CC2CO)=O)c1C C1(CC=C)(NC(=O)CCS(=O)(=O)NC)CCN(C(C2CC2C#N)=O)CC1 CC1(C(=O)NC2CCCC2NC(=O)C(F)Cc2ccccc2)CC=CC1 C1(NC(CCCNC(C)=O)=O)CC2CCC1N2C(c1nc(C)sc1C)=O [N-]=[N+]=NCCC(=O)NCc1occc1C(=O)N(C1CCCC1O)C1CC1 N1(C(C2CC(CCC)OCC2)=O)CC2CC(NC(=O)Cn3ccnn3)C2C1 C1(NC(c2scc(C)c2Cl)=O)CC2CC(C1)N(C(=O)C(C)OCC(C)C)C2 N1(C(C=C(C)Cl)=O)CCCC1C(C)NC(=O)C(C1CCOCC1)O C(=O)(C(CC)C(C)C)N1CCCC(CN(C(=O)CCc2cc(C)[nH]n2)CC)C1 N1(C(C(CC=C)C)=O)C(CNC(=O)Cc2cccc(C)c2Br)CC2CCCC12 CCCC(CNC(c1ccc(C)c(C)c1)=O)C(=O)NCC(C)CCCO CC1=CCC(C(=O)NC(C)CC(C)NC(C2C3CCC2CC3)=O)CC1 c1(C(=O)NC2CC2CNC(C2CCCN(CC(F)F)C2)=O)ccc2cc[nH]c2n1 N1(C(c2c(OCC)nccc2)=O)CCCC(CO)(NC(=O)CCC2CC2(Cl)Cl)C1 N1(C(C2CN(C(C)=O)C2)=O)CCC2(CC1)CN(C(C1(C)CC1F)=O)CCO2 N1(CC(=O)NCC(CCNC(CN(C(COC)=O)C)=O)O)Cc2ccccc2C1 c1(CN)cnc(C(=O)NC(c2ccccc2)CC2CCOC2)cn1 N1(C(c2c(C)cc[nH]c2=N)=O)CCC2(CCN(C(=O)CCCn3cncn3)C2)C1 C(=O)(CCCCC1CC1)NCC1CC(CNC(=O)CCn2ccnn2)OC1 N1(C(c2cc(N(C)C)ncc2)C(=O)NC2CCOC2)CC(C(F)(F)F)CC(C)C1 C1(C(N2CC(NC(C(C(C)C)N(CC)CC)=O)C2)=O)CCC2(CCCO2)CC1 C(CCC(C(=O)NCCC(=O)NC1CC1)NC(c1nccnc1N)=O)OC CC1CN(C(=O)C(C)(C)c2cnco2)CC(C)N(C(=O)CCc2ncc[nH]2)C1 S(=O)(=O)(c1ccc(N2CCC(C(C)C)CC2)cc1Br)N(CC(CC)O)CC1CC1 c1(C(=O)NC2C3(CCN(c4nccc(C)n4)CC3)C2)cc(F)c(F)c(Cl)c1F N1(C(c2c(CCC)[nH]cc2)=O)CC2COCC2(C(N2CCCCCCC2)=O)C1 c1(C(=O)N(C2(C(=O)NCC(C3CCC3)C3CC3)CCC2)C2CC2)cc(F)c[nH]1 c1(CC)ccc(CN2CCSC(C(=O)Nc3cccc(F)c3CO)C2)cc1C CC1OCCCC1C(=O)N(O)Cc1cn(C2CCOCC2)nn1 C1(NC(COCCC=C)=O)CCN(C(=O)Cc2cc(C)cs2)C12CCC2 c1(CC(C)(C)NC(Cc2nc(C)nn2C)=O)c[nH]c2ccc(Br)cc12 C(=O)(C(C)(C)C1=CCN(C(=O)Cc2cc[nH]n2)C1)NC1C(C)COC1 C(=O)(CCCN=[N+]=[N-])NC1CC(CNC(C2CC(CC)C2)=O)C1 N1(C(C2CN(C(Cc3cc(C)no3)=O)C2)=O)CC2CCCC2C12CC2 N1(C(C2CCN(C)CC2)=O)CCC(F)(F)C(CNC(c2cnc(S)[nH]2)=O)C1 c1(N2CC(C)C(C)C2)ncnc2c1ncn2C(CO)C1(N2CCCC2)CC1 c1(CC(=O)NC2C(OC)CN(C(C=C(CCC)C)=O)C2)cc(Cl)ccc1OC Cc1ccccc1Cn1cnc(NC(=O)CCc2cn(-c3ccccc3)nn2)n1 N1(c2n(-c3ccc(C)cc3)nnn2)CCN(C(=O)C2CC2)C(C#N)C1 C1(N(C(c2cc(C(=O)OC)ncc2)=O)C)CCCN(C(=O)Cn2ncnn2)CC1 C1(O)(CC(=O)NC2(C3CCCN3C(c3cncs3)=O)CC2)CCCC1 c1(NC(C2CCCNC2)C)cc(NS(=O)(=O)Cc2ccccc2)nc(C)n1 c1(C(=O)NC2(C)CN(C(Cn3nc(C)n(C)c3=O)=O)C2)cccc2c1ccn2C C1(C)(CNC(C(C=C)O)=O)CCCN1C(=O)CCCCN(C)C c1(CC)cc(F)ccc1C(=O)NC(C)(CNC(C1CCCN1N=O)=O)C1CC1 C12(N(c3cc(Br)n[nH]3)C(=O)N(C)C)CC3CC(CC(C3)C1)C2.C=C1CNCC1 N1(C(c2cnn(CCCC)c2C)=O)CCCC(O)(CNC(=O)CCC2CC2C)C1 c1(N2CC(C)(CNC(C(C)(C)SC)=O)OCC2)nc2ncc(Cl)cc2o1 c1(C(=O)OC)cccc(C(N2CCOC(CCNC(=O)CCC=C(C)C)C2)=O)n1 C(=O)(C(F)C(=O)N1CCCC1C(C)NC(=O)CC1CCCOCC1)OCC c1(C(=O)NC(C2CCN(C(c3c[nH]nc3F)=O)C2)C)cc2cccc(Cl)c2[nH]1 C(=O)(C1=CCC(C)CC1)NC(C1CCN(C(c2ccc3n[nH]cc3n2)=O)CC1)C c1(C(N(C(C)C(=O)NCC(O)COC)CC#C)=O)ccc(C#C)cc1C C1(C(N2C(CNC(COC(CC)(C)C)=O)CC(O)C2)=O)CCC(N=[N+]=[N-])CC1 O(N=C1CCCCCC1)CC(=O)NCC(C)N(C)C(c1csc(Br)n1)=O C1(NC(C(C)NS(CCCC)(=O)=O)=O)CCN(C(=O)CCCOC(C)=O)CC1O Cc1cc(C(=O)NC2C3CC4C2C4C3C(=O)Nc2cncc(CO)c2)ccc1F c1(CNC(CCC=C)=O)ccc(N2CCN(C(C3CNCCO3)=O)CC2)cc1 C1(C)(C(N2CC(O)(CNC(C3CCC(NC(CC)=O)C3)=O)C2)=O)CNC(=O)C1 c1(C(=O)NC(CNC(CC(C=C)C)=O)C2CCC2)ccc(Cl)c(Cl)c1O Cc1ccc(Cl)c(OCC(=O)NC2CCC(CNC(=O)C(F)=C3CCC3)CC2)c1 CC1NCCC1CCNC(=O)Nc1cn(C)nn1 CC1(C)COC(C(=O)NC2CCN(C(c3ccc(C(C)(C)C)[nH]3)=O)C2)C1 O=C1COc2ccc(S(=O)(=O)N3CCC(CCO)C3)cc2N1 c1(-n2cc(C(CC)N(C)C)nn2)ccc(CCNC(c2sncc2Br)=O)cc1 CN(CCCC(=O)N1CC2CC1C2NC(C1CCCCN1CC(F)F)=O)N=O c1(OCCOC)cccc(C(=O)NC(C)CNC(C2C3COCC23)=O)c1 C1(COC(CNC(C2(C(=O)NCC(C)C)CC2)=O)=O)CCCC1.C(C)(=O)O c1(CC)ccc(C(N2CC(CN(C)C(c3scnc3COC)=O)C2)=O)c(F)c1 C(C(=O)Nn1cccn1)NC(C(C)=CC(C)(C)C)=O N1(C(c2c(CC)cno2)=O)CC(N(C(=O)CC2OCCC2(C)C)C)C(C)(C)C1 CCC(CCC(=O)NC1CC(O)C(F)C1)NC(=O)Cc1ncoc1C c1(CN2C(CNC(c3n(C)ccn3)=O)CCC2)ccccc1Cl N1(C(c2occc2Br)=O)CCOC2(C1)CN(Cc1sccc1Br)C2 C(=O)(C1CCc2c[nH]nc21)NCCCCNC(C1CCC(C2CC2)CC1)=O C(=O)(C(O)CCC(C)C)NCC1(C)CCN(C(c2cnnc(C)c2C)=O)C1 C1(CNC(CC(CNC(=O)CC(=O)N(C)C)OC)=O)OCC2CCC1C2 N1(C(c2c(C)cc(Br)cn2)=O)CCC(NC(=O)C=CCO)CC(C)(C)C1 c1(C2c3nc2cs3)cn(CCCF)nn1.CC(C(=O)O)N(C(=O)CN(C)C)C N1(CCOCC)CC2CCC(C1)O2.c12cccc(c1)C1CCCN1C2 C1(C)(CNC(CCC(C)SC)=O)CC(F)(F)CN1C(=O)C1=NNC(=O)CC1 N1(C(c2nc(C)sc2)=O)CCC(O)C1C(=O)Nc1cnns1 N#Cc1ccc2c(NC(C3CC3C(=O)Nc3cc(Br)cc(Cl)n3)=O)n[nH]c2c1 CC(C)C(C(=O)NCC=C1CCN(C(C2C3CCOCC23)=O)CC1)NC=O C1(NC(C(C2CC2)OCC)=O)CC2CN(C(c3ncc(F)cn3)=O)CC12 c1(C(=O)NCC2CN(C(C(C(=C)Cl)(C)C)=O)CC2(C)C)ccc2c(c1)CCOC2 C1(C(=O)NCC2N(C(C3OCCN(C)C3)=O)CCCC2)CCC(C)(C)CC1 C(=O)(C(C)(C)CC(=O)NC(C)C(C)NC(=O)CC(C)(C)OC)OC C12(NC(c3ccc(OC(F)F)cn3)=O)CCN(C(c3ccsc3)=O)CC1C2 N(C(=NCCC)NCC(c1cccs1)N1CCCC1)C(C#C)CCC c1(C(N2CC(CNC(C(CC)F)=O)N(C)CC2)=O)sc2[nH]c(C)nc(=O)c2c1C C1(C)(C(N2CC(C)C(NC(c3ncc(F)cn3)=O)C2)=O)CCNC(=O)C1 N1(C(CC(C)O)=O)CCN(C(c2ccc(C3CC3)cc2F)=O)CC1CC(F)(F)F N1(C(Cc2cccc(OC)c2)=O)CCCC2(CCCN2C(c2cccn2C)=O)C1 CCC(CC(F)(F)F)C(=O)NC1CN(C(C2CC3(CCC3)C2)=O)CC1C CC(O)CCCCCC(=O)N1CC2(C1)SCCC2NC(=O)C#CC1(C)COC1 C(CC(=O)N(CC(C)(C)COC)C)(CC(C)C)NC(c1cc(CC)on1)=O c1(CCC(=O)NC2CCN(C(COCC)=O)CC2O)cc2ccccc2nc1O N1(C(C2ON=C(C)C2C)=O)CCC(O)C(NC(=O)Cn2ncc(Cl)c2C)C1 N1(CC=C(C)C)CCN(C(c2c(CO)noc2C)=O)C(C)C1 c1(C(=O)NCCCN(C(=O)CCC2CCC(=O)N2)CC)cncn1C(C)C C1(NC(c2coc(Cl)n2)=O)CC2COCC(C1)C2NC(C1CC(C(F)(F)F)C1)=O CN1CCC(NC(=O)C=Cc2cn[nH]c2)C12CCCN(C(c1nn[nH]c1Cl)=O)C2 Cc1cc(CNC(=O)CC2CCC(NC(=O)CC3CC(F)(F)C3)C2)n(C)n1 C1(C2(NC(c3ccc(C4CCC4=O)cc3)=O)CC2)(OC)CCC1 C1(C(N2CCCC(CN(C)C(C3CCCCO3)=O)C2)=O)CCCCC1(F)F N1(C(C(C2(OC)CCCC2)(F)F)=O)CC2(COC(CNC(=O)C(C)N(C)C)C2)C1 c1(C(=O)NC(c2n(C)ncc2)CNC(C2CC23CC3)=O)[nH]cnc1C#N C(=O)(N1CC(C(=O)NC(C)(C)CNS(=O)(=O)N(C)C)CC(=O)N1)OC(C)(C)C C1(C(N2CC(C(N(C)CCO)=O)OCC2)=O)CC(=O)CC12CCC2 Cc1n[nH]cc1C(=O)NCCC1CN(C(C2(c3cccs3)CC2)=O)C1 c1(CC)ccc(CN2CC3CC(C2)N3C(c2cc(Br)cnc2C)=O)c(O)c1 n1(CC)cnnc1C(=O)NC(C)CCCNC(C1(CS(N)(=O)=O)COC1)=O C(=O)(C(C)(C)CNC(c1cscc1Cl)=O)NC(C)Cc1nc[nH]n1 c1(C(=O)NC2CN(C(CCCc3ccc(CC)cc3)=O)C2)cc(N)nc(Br)c1 Cn1ncc(C(=O)NC2(CCCNC(=O)CC3CC(F)C3)CC2)c1S(N)(=O)=O N1(C(C2CCN(C)C2)=O)CC(NC(=O)Cc2cccnc2O)CC(C)(C)C1 c1(OC)cccc(C(=O)NCC2(CN(C)C(C3CCC(F)(F)C3)=O)CC2)c1N N1(CC(=O)NCC2C(NC(c3ccc(C(N)=O)[nH]3)=O)CC2)CCS(=O)CC1 c1(C(N2CCN(C(CNC(CC3(C)CCOC3)=O)=O)CC2)=O)ccnc2c1CCC2 n1(CCCC(=O)NC2CC(F)(CNC(C3C(C)CCC3)=O)C2)cnc(C#N)n1 C(=O)(C1=CCN(C(=O)C(C(C)C)N(C)C)C1)NC(c1ccc(C)cn1)C c1(-c2cc(C)cc(O)c2)cnn2cc(C(=O)Nc3cc(F)c(C)c(Br)c3)cnc12 C1(CNC(c2scnc2C(F)(F)F)=O)CC(F)(F)CN1C(=O)C=CC1CCCO1 C1(C(N2CC(C)(C)OCC2CNC(c2cnc[nH]2)=O)=O)Cc2ccccc2O1 C1(NC(c2c(OC)oc(C)n2)=O)CN(C(C2(C)CCC(=O)N2)=O)CCC1CO c1(CNC(c2nnnn2CCSC)C2(CC)CC2)ccc(NC)cc1 C1(N(C(COC)=O)C(=O)Cc2cc(F)ccc2Br)COC2(CCNCC2)C1 c1(-c2nc(CCCC)nn2C2CCOC2C)ccc(CO)c(C(C)C)c1 c1(NCC(CNC(c2c(C(C)C)n[nH]c2)=O)O)cc(O)nc(O)n1 N1(C(c2n(C)cc(C#N)c2)=O)CCNCC12CCOCC2 c1(C(C)NC(CC(=O)OCC)C)cc(F)c(OC)c(F)c1 C(=O)(CCCCCCNC(c1cc(C2CC2)no1)=O)N(C1CCCCC1)CC c1(C(N2C3C(NC(C4CCC4)=O)(CCC3)CCC2)=O)cnc2ccccn2c1=O N1(C(C(C=C)O)=O)CCCC(C2CCN(C(C3(C4CC4)CCCO3)=O)CC2)C1 O=C1CNC(=O)C(CC(N2CC(NC(c3cc4c(s3)CCC4)=O)C(O)C2)=O)N1 C(CCCCN1CCCC1)(C(=O)O)NC(c1c(CC)n(CC)nn1)=O C1(C(C(=O)NCC2CCCO2)N(C(C)CC#N)C)CCC2(CC1)CC2(F)F C(=O)(C(C)(C)C(C)(F)F)NCCN(C)C(c1ccn(-c2ccccc2Cl)n1)=O c1(C(=O)NCCOC2CN(C(C(C(C)C)OC)=O)C2)cnc2nc(Cl)ccc2c1 C(CNC(c1cnn(CCNC(=O)C(F)=CC2CC2)c1)=O)(C(C)(C)C)OC C(C(CC(=O)NCCC1CC(F)(F)C1)C1CCC1)NC(c1c(C)csc1)=O C1(NC(C2N(C(C)=O)CCC2)=O)CCN(C(=O)C(C)(C)CN(C)C)CC1CC1CC1 C1(NC(CNC(C(CC)C)=O)=O)CC(F)CN(C(=O)CN2CCOCC2)C1 C=CCCCCCC(=O)N1C(C(=O)NCC2(C)CNC(=O)O2)CCC1C1CC1 Cc1cccc(C(=O)N(C)CC2CN(C(=O)C(C)NC(C)(C)C)C2)c1F N1(C(c2csnn2)C)CCN(C(c2ccncc2F)=O)C(C)C1 c1(OC)ccc(C(=O)NCc2ccc(Cl)cc2C)cc1OCCN(C)C c1(C(=O)NC(C)CNC(=O)CC(C)(C)C(F)(F)F)cc2c(cc1[N+](=O)[O-])OCO2 N1(CC(N2CCOCC2Cc2cccc(Cl)c2)=O)CCc2ccccc21 CC(C)S(=O)(=O)C(C)C(=O)NCC12CC1CN(C(c1cc(F)c[nH]1)=O)C2 N1(C(C(CC)(C)F)=O)CCN(C)C(CNC(=O)Cc2ccc(F)cc2F)C1 O=C(NOCC(O)C(F)(F)F)C(O)CNC(=O)Cc1cccnc1F CC(CC(C)C(F)F)NC(=O)CC1CCN1C(c1sccc1C#N)=O N1(Cc2c(C)c3c(o2)cccc3)CCC2(CC1)CN(C(c1ccsn1)=O)CCO2 C(CNC(C1CC(C)CO1)=O)(CCNC(C1CC(F)(CF)C1)=O)OC C1(NCc2ncn(-c3ccccc3)n2)CC2(C1)CC1CNCC1C2 n1(CC(=O)N(CCC(=O)NC2(C(=O)NCC)CC2)CC2CC2)ccc(C)c1 c1(C(N2CCCCC(NC(C3CC(CCC)C3)=O)C2)=O)ccc(S(C)(=O)=O)cc1 Cc1nc(NC2CC2)sc1C(=O)NCC(CO)NC(c1ccc(C(N)=O)cc1)=O C1(CCC)CCCCC1NC(C1(NC(=O)NC2CC(CO)C2)CCOCC1)=O Cc1[nH]nc(C(N2CC3C(CNC(=O)Cc4cccc(F)c4)C3C2)=O)c1Cl N1(C(c2ccc(C)cc2O)=O)CC2CC(C)N(C(c3cc4ccsc4s3)=O)C2C1 C1(C(=O)NC(C)CCCNC(=O)Cn2ncnn2)C2CCC1CC2 N1(C(CC(CC)(F)F)=O)CC2CC1CCN2C(=O)CSCCC(F)(F)F N1(C(c2ccc(CCC(=O)OC)s2)C(=O)NCC(=C)C)CC(C)S(=O)C(C)C1 C=C(C)CCC(=O)NCC(O)CNC(=O)Cn1nc(C)cc1C(F)F C1(c2nnnn2C2(C)CC2)(NCCC(=O)OC(C)C)CN(C(C)=O)C1C CCC(C)CCCC(=O)NC(C)C(C)C(=O)N1CCOCC1 C1(CNC(Cc2c(C)noc2C)=O)CN(C(=O)Cc2cncs2)CCCO1 c1(N2CC3(CN(C(CCCSC)=O)C3)C2)c(C#N)cnc2ccc(Cl)cc12 C(=O)(C1CC(=O)Nc2ncn(C)c21)NCC1(O)CCCN(C(C2CC(C)C2)=O)C1 N#Cc1ccccc1NC(C12CC(C(=O)NC3(c4ccccc4Cl)CC3)(C1)C2)=O c1(C(N2CCC(CCNC(C(C)OC(C)(C)C)=O)C2)=O)cn(C)nc1C(C)(C)C C1(CNC(c2cccc(=S)n2O)=O)CN(C(c2cc(O)ncn2)=O)CC12CCC2 C(C)(C)(CC(F)C(=O)NCC(O)CCO)NC(c1c(C)c(O)ccc1)=O C(CCCCC=O)N(C(CCN(CC)CC)=O)CC.C(C(C)CO)NC CCC(C)CCCC(=O)NCCSCC(=O)NCC(C)(C)C#N C1(CCCC)CN(C(=O)CN2CCSCC2)CCN1C(C12COCC1C2)=O N1(C(c2ccccc2)C(=O)NCC=C)CCOCC(C(=O)OC)C1 c1(C(N(C2CCCC2)CCNC(=O)CN2CC3CC3C2)=O)ccn(CO)c(=O)c1 N1(C(C(C2CCC2)OCC)=O)CCC(C2CC2NC(=O)C=C(C)C(C)(C)C)CC1 c1(CC(=O)N(CCNC(Cc2nnc(C)o2)=O)C(C)C)cn2cccc(C)c2n1 CC1CN(C(c2cnc(O)s2)=O)CC1(C)CNC(=O)C(C)(C)n1cccn1 N1(C(c2c(OCCC)ccc(Cl)c2)=O)Cc2ccc(CO)cc2C1 C#Cc1cccc(C(=O)NC(C)(CC)CCNC(=O)C(CCC)OCC)c1C N1(C(C(C2CCC2)OC)=O)CC2CC1C2NC(=O)CC(C)(C)C1CCC1 c1(C(=O)NCC2CC(C)N(C(c3c[nH]ccc3=N)=O)C2)ccc(C(F)F)cc1F N1(C(CC=C)=O)CCc2cc(C(=O)Nc3ccc(C#N)cc3)ccc2C1 c1(N(C)C)nc(C(=O)NCC(F)CNC(=O)CCS(C)(=O)=O)cc(O)n1 c1(NC(=O)NCc2cnc(C(C)(C)C)nc2)c(Cl)ccc2c1CCO2 c1(OC)cc(-c2cn(CC(=O)NCc3sc(C)cc3Br)nn2)cnc1O.C1CC1 c1(NC2C=CC(C(=O)OC)C2)ccccc1CC(=O)NC(C)=O c1(C(N(CC(C)CNC(c2cnco2)=O)C)=O)cccc(CS(C)=O)c1 Cc1cccc(CS(=O)C(C)C)c1F CC(C)CC(F)C(=O)NC1CC2(C1)CC(NC(c1sccc1-n1cnnn1)=O)C2 c1(C(N2CC(CC(C(N3CC(C#C)(F)C3)=O)F)C2)=O)ccc(NC)c(F)c1 C1(NC(COCc2onc(CC)n2)=O)CN(C(c2ccncc2C)=O)C2CC12 N1(C(C(C)NS(C)(=O)=O)=O)CC(C(N)=O)(CNC(C2CC(F)C2)=O)C1 C1(NC(c2c(C)nn(C(C)C)c2)=O)CC2CC1CN2C(=O)CCc1nc(O)n[nH]1 c1(C(=O)NCCn2ccc(C(N3C(CN(C)C)CCC3)=O)c2)cc([N+](=O)[O-])c[nH]1 c1(CCC=C)cccc(C(=O)NC(C)CC(C)CC)c1 c1(OC)c(N2CCOCC(NC(c3cn4c(n3)CCC4)=O)C2)ncnc1Cl N1(C(C(C)C2CCOC2)C(=O)NCCC2CC2)Cc2cccc(F)c2C(C)(C)C1 N1(C(C(CC)C#N)=O)CCCC(C(=O)NCC(O)CCOC)(CC)C1 C1(CNC(CN(C)C(c2ccsc2)=O)=O)CN(C(c2cncc(F)c2)=O)CCN1C c1(C(=O)NCc2cc(C(N(CCOCC)C)=O)n[nH]2)nn(C)cc1Cl C12(C(N3CCC(C)C3)=O)CCC(CC1NC(=O)CC1=CCCC1)C2 N1(C(c2cncc(NCC)c2)=O)CC(NC(c2cccc(=O)o2)=O)C(C2CC2)C1 C12(C(=O)NCC(O)COc3ccccc3)CCCC1NCC2 C1(CNC(C2CN(C)C2)=O)CN(C(c2nn[nH]c2Cl)=O)CC12CC2 N1(C(C(c2cn(C)nc2)O)=O)CC(F)(F)CC1CCNC(c1ncc(F)cn1)=O S(=O)(=O)(C1CN(C(C2C=CCCC2)=O)C1)N1CCN(C(=O)C(F)C2CCC2)CC1 C1(F)(CNC(C2CCCC2(F)F)=O)CCN(C(c2nn(C(F)F)cc2Cl)=O)C1 c1(CN2CC(ONC(c3occ(C(=O)OC)c3)=O)C2)cn(C)cc1C C(=O)(C(C(CC)CC)N(C)C)N1CCN(C(COCCSC)=O)CC1CO C1(CNC(C2ON=C(C)C2)=O)C2CN(C(c3c[nH]nc3Br)=O)CC12 C(=O)(C(C)(COC)CC)N1CCC(C(C(=O)NC(CCC=C)C)C)CC1 Cc1cccc(Cn2cc(C3(C)CCCN3C(=O)COC(C)C)nn2)c1Br Cc1cc(C(F)F)oc1C(=O)NCC1(NC(=O)C=Cc2cccn2C)CCCC1 N1(C(CCCN(C)C)=O)CC(CNC(=O)C(C)(C)N(C)C)C(c2cncn2C)C1 CC1(C)C(C)(C)C1(F)C(N1CCC(O)(CNC(C2CC3(C2)CC3(F)F)=O)CC1)=O C(=O)(C(C)(F)CC)NCC(CC)NC(=O)C(=O)NCCC(N)=O Cc1ccc2c(n1)OCCN2C(=O)C(O)C(F)(F)c1ccccc1 Cc1cc(C(=O)NCCn2cc(C(=O)NC3CN(C)CC3C)nn2)c(C)s1 N1(C(c2cccc(C)n2)=O)CC2(CO)CC1(C(N1C3CCC1CC3)=O)C2 C1(Nc2n(C)ccc(=O)c2)C2CC3CN(C(=O)OC(C)(C)C)C1C3C2 c1(OC)ccc(Br)cc1C(=O)NCC(N1CCC(NC(=O)CCOC)C1)=O N1(C(C(C)NC(C)=O)=O)CC(NC(=O)C(c2ccc(Br)cc2)(C)C)C(C)C1 CC1CN(C(C2CC(CC(C)(C)C)C2)=O)CCN1C(C1CCOCC1)=O Cc1csc(C=CC(=O)NC(CO)C(C)NC(=O)C=Cc2nccs2)n1 c1(C(=O)NC2C=CCN(C(CCC=C)=O)C2)ccc2nnc(O)n2c1 N1(C(C(C)OCCCC)=O)C2CCC1CN(C(C1(C3CC3)CCOCC1)=O)CC2 c1(COC(C(=O)NC2CCC(CNC(C(C)NS(C)(=O)=O)=O)C2)C)ccccc1 Cc1ccc(C(=O)NCCCCC(C)NC(=O)CCOC2CCOC2)c(F)c1Cl C1(Nc2nccc(OCC)n2)CS(=O)(=O)CC1NC(=O)C(F)(F)C(F)F C1(CNC(C2ON=C(C)C2)=O)CC(NC(=O)C=Cc2ccsc2)CCO1 CC(C)CC(C)CC(=O)NCCCNC(c1cc(CS(C)(=O)=O)on1)=O C1(CC)CN(C(C2CC2F)=O)CCN1C(=O)Cc1ccsc1C C(=O)(CCC(C)NC(c1cccc(CC#N)c1)=O)NC(C(CO)SC)C c1(CC(C)C(=O)NC(CNC(=O)CC23CCC(CC2)C3)CO)ccc(F)cc1 CC1CC(CNC(C2CC2C(C)O)=O)CN1c1ccnc(Cl)n1 C1(NC(=O)CNC(N2CCCC2)=O)CC12CCC(NC(C1(C(F)F)CC1)=O)CC2 N1(CC(N2C(C)CC(NC(=O)CCc3nccs3)C2)=O)C(=O)NC(C)(C)C1=O c1(C(N(CCOC)CCNC(C23CCCCC2C3)=O)=O)ccc(C2CC2)nc1C C1(C)(C(N(CC(CC)OC)C)=O)CCCN(C(=O)CSc2cccc(Cl)c2)C1 C(=O)(CC(C)(C)CNC(C1COCCC1C)=O)N(CCOCC=C)C C(=O)(C1=CCCCC1)N(C1CCCC1)CCNC(C(C)(C1CC1)OC)=O c1(C(N2CC(C(=O)Nc3c(C(=O)OC)nsc3)SCC2)=O)ncc(Br)cc1F CCC(C)C(C(=O)NCCCOCC(C)C)N(C)C(c1csc(Cl)c1)=O N1(C(c2nc(-c3cn(C)nc3)sc2)=O)CCC2(CCN(C(=O)C(C)(C)F)C2)C1 c1(CC(=O)NCC(CNC(c2cc(COC)no2)=O)O)cc(C)cc(Br)c1 Cc1c(C(N2CC(C(C)NC(C3CCC4CC34)=O)C2)=O)ccn1C(C)C c1(C(=O)NC2(C)CN(C(CC3CC(OC)C34CCC4)=O)C2)cccn2cncc12 N1(C(C2(C=C)CCC2)=O)CC(NC(=O)CN2CCC(C)C2)C(C)C1 C(=O)(C1=CC(C)CC1)N(CCC)CCNC(c1ccc(SC(F)(F)F)o1)=O N1(C(CCOC(C)=O)=O)CCCN(C(=O)C(C)Cc2cccnc2)CC1CO C1(S(C)(=O)=O)(C(N2CC(CCC)N(C(=O)Cc3ccns3)CC2)=O)CCOCC1 Cc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCCC3N)cc1C c1(COC(C2(C)CC(C3CC3)=NO2)=O)nc(=N)[nH]c(=Nc2ccccc2)[nH]1 Cc1cc(C(=O)NCC2CCCN2C(C2CCOC2)=O)nc(N(C)C)n1 c1(CN2CCC(N(C)C(c3nc(Br)ccc3F)=O)C2)c[nH]c2cc(Br)ccc12 c1(C(N(CC(CC)NC(=O)CC2CC3(COC3)C2)CC)=O)ncc(Cl)cc1Cl C(=O)(C(CC(C)C)NN1CCSCC1c1noc(Cc2ccccc2)n1)OCC C(=O)(CCCCCN(C)C)NCCC(C)NC(C1(C)CCCN1C)=O CC1(C)CCCC(C(=O)NCC2(NC(c3coc(Br)n3)=O)CCC2)CC1 N1(C(c2ccc(C)o2)=O)CCCC(C)C1C(=O)NCc1c(C(C)C)cccc1F c1(C(N2CC(N(C(CSCC)=O)C)C3(C2)CC3)=O)cnc2ccc(C)cc2c1 c1(-c2ccc(NC(C3(CC)CCOCC3)=O)nn2)ccnc(C#N)c1 c1(CC(=O)NC2CCC(NC(=O)C=Cc3cn[nH]c3)CC2)ccc2ocnc2c1 N1(CCOCC)CC2CCC1CN2C(=O)Cc1ccoc1 C1(NC(C(C#C)(C)C)=O)CCCN(C(c2ccc(Br)cc2OC)=O)CCC1 C1(NC(CCCC)=O)CN(C(C2CCCCN2C(=O)Cc2cccs2)=O)CC1O CSC=CC(=O)NC1(CCNC(=O)C(C)Cn2cccn2)CCCC1 N1(C(C=CCC)=O)CC(CNC(c2noc(-c3cccc(Cl)c3)n2)=O)C2(CC2)C1 Cc1cc(C(N)=O)cc(S(=O)(=O)NCCNC(=O)C=CC2CCOC2)c1C Cn1cnc(=NC(=O)NC2(Cc3ccc(Cl)c(F)c3)CC2)[nH]1 Cc1cnccc1C(N1CC2C(NC(c3cccc(NS(C)(=O)=O)c3)=O)C2C1)=O C#CC1(C(=O)NCC(CC)NC(=O)C(c2ccc(F)cc2)N(C)C)CCCC1 C1(CNC(C2(CCC=C)CCCC2)=O)COCCN(C(=O)CCOC(C)C)C1 c1(C(CSC)NC2CC(C(F)(F)F)CC(c3ccccc3)C2)ccc(F)cc1F S(=O)(=O)(C1CCC(C(F)(F)F)CC1)NCC1(C)CCOC1C1CC1 c1(C2CCN(c3nnc(C(=O)OC)s3)C2)ccc(Br)cc1 c1(C(N2C(CNC(c3c(C)cccc3F)=O)C(C)CC2)=O)cc(O)cc(Cl)c1Cl N1(C(CNC(CC)=O)=O)CCCC2(C1)CN(C(c1c(C)nn(CC)c1Cl)=O)C2 Cc1oc(S(C)(=O)=O)cc1C(N1CCCCC1CNC(=O)Cn1cnnc1O)=O c1(CCC(=O)N(C)CCN(C(=O)Cc2cnc[nH]2)C)cc(Cl)sc1Cl C#CCCCC(C)C(=O)N1CC2CC1(C(N1CC(F)(F)CC1CO)=O)C2 c1(C(O)Sc2ccc(-c3ccc(C(C)C)cc3)cc2)ccc(Cl)c(F)c1 CCC(C)C(C(=O)NC(C1(C(=O)N(C(C)CN(C)C(C)=O)C)CC1)C)N(C)C CCC(CC)C(=O)NC(CCNC(C1(OC)CCC1)=O)C(C)C CC1(C)CCCCC(C(N2CC3CC(C2)N(C(=O)C(O)CC(N)=O)C3)=O)C1 N1(Cc2c(CC)cccc2)CC(F)(F)CC1C(N1CCCC1C(=O)OC)=O c1(CN2CC(C(=O)Nc3ccc(C(C)(C)C)nc3)C2)c(C(F)(F)F)cccc1O c1(C(N2CCC(N(C(C(C3CC3)OCC)=O)C)C2)=O)c(O)ccc(Cl)c1O N1(C(C(C(C)C)C)=O)C2CCC1CC(NC(c1cccc(Cl)c1)=O)C2 N1(C(C2=NOC(C)C2)=O)CC2OCC(NC(c3csc(C(C)(C)C)c3)=O)C2C1 C=CC1CCCN1C(C1(CCNC(c2cn(C3CC3)nn2)=O)CCC1)=O CC12COCC1(C)CN(C(C1CCCC1NC(c1ccsn1)=O)=O)C2 c1(C(=O)NC(CCCNC(C(C)OCC)=O)C)ccc(Br)nc1N N1(C(CC(=C)C)=O)CCCC(CO)(CNC(c2cccc(F)c2F)=O)C1 c1(NC(C2CCCCN2Cc2cc(Cl)nc(Cl)c2)=O)ccc2ncnc(O)c2c1 c1(OCC)ccc(NCc2nnnn2C2CCCC2)cc1.C(C)(CCOC)N CC1(C(=O)NCC2CC(NC(C3CSC3)=O)C2)CCc2ccccc21 C1(NC(=O)CCF)CC12CCC(NC(=O)Cc1ccc(F)c(Br)c1)CC2 c1(C(N2CCN(C(c3ccc(O)nn3)=O)C(CO)C2)=O)ccc(Cl)c(O)c1 C1(COC)(NC(=O)C(CO)N(C)C)CCCN(C(=O)C=CC2CCCCC2)C1 N#Cc1ccc(C(N2CC=CC(NC(=O)CC3CCCN3C(N)=O)C2)=O)cc1 c1(C(=O)NC(CN(C(=O)CCP(C)(C)=O)CC)C)c(C)[nH]c(C(=O)OC)c1C c1(CCC(C)Nc2c(NCC)cccc2)nc2ccccc2[nH]1 N1(C(c2c(N)c(F)ncc2)=O)CC2=C(C1)CN(C(=O)CCC1CCCO1)C2 N1(C(C(C)OC)=O)CCC(C(C)NC(=O)CNC(c2cccs2)=O)CC1 c1(C(=O)NC2CN(Cc3c(C)nc[nH]3)CC2F)ccc(CO)nc1 C1(CCNC(c2n(CCCSC)nnn2)c2ccns2)CCc2ccccc2C1 N1(c2c(C(=O)OC)cccn2)CCC(NC(=O)CSS(C)(=O)=O)CC1C N1(C(c2c(C)cccc2F)=O)CC2CN(C(=O)CC34COC(C)(C3)C4)CC2C1 CCCC(C)(CCC)C(=O)N1CCC(C(C)NC(c2cc3ncccc3o2)=O)C1 NC1CC2CCC(C1)N2C(=O)Cc1cccc2sccc12 N1(C(C(C=C)(C)O)=O)CCc2c(C(=O)NCC3CCOC3)cccc2C1 N1(C(CS(=O)(=O)N(C)C)=O)CCC2CCCC12CNC(C1(C)CS(=O)(=O)C1)=O C(=O)(C(C#N)C(C)(C)C)NC1CC(CNC(c2nn(CC)c(=O)cc2)=O)C(O)C1 C1(C(N2CC(CNC(=O)CN3CC4CC4C3)C2)=O)CN2CCCN1CC2 C(C(CC(F)(F)F)NC(C1CCCCC(=O)N1)=O)NC(C1(CC(C)C)CC1)=O C#Cc1cccc(CC(N2CCC(F)C(NC(C3CN(C)CCO3)=O)C2)=O)c1 C1(C=O)CC2(C)CCC1(C)O2.C1(NC)CN(C(C)C)C1 C1(C(N2CCN(C(c3cncc(C)n3)=O)C(C)C2)=O)(OCC)CCCCCC1 C(N=c1nc(-c2ccccc2)nc(N2CCOC3(CCC3)C2)[nH]1)C1(C)CC1(F)F c1(NC(C2N(C(CCC(=O)OC)=O)CC3C2C3(C)C)=O)ccc(Br)nc1[N+](=O)[O-] Cc1cc(Br)cc(C(N2CCN(C(C3CCCN3C)=O)CC2C(F)F)=O)c1C c1(C(=O)NCCOCCN(C)C(C2C(C(F)F)C2(C)C)=O)csc(C2CC2)n1 C(CN=c1cc(NC(C)Cc2ccc(C)cc2)nc(C)[nH]1)N(CCO)CC N1(C(C2C(C=C)CC2)=O)CCCN(CCNC(=O)CCc2nnc(C)n2C)CC1 c1(C(N2C(C(N(C)CC3CCCC3(C)C)=O)CCOCC2)=O)ccc2cccnn12 N1(CC(C)C)CCN(C(C2CCN(C(C3CCSCC3)=O)C2C)=O)CC1 N1(C(C2N(C)CCOC2)=O)CCCC(NC(c2ncoc2C2CCCO2)=O)CC1 Cc1cc(C(=O)NCC2(F)CCN(C(=O)CCC=CC(C)C)CC2)cc(N)c1 N1(C(CCNC(=O)OC(C)(C)C)=O)CC2CCC1C(NC(c1ccc(Cl)s1)=O)C2 C1(C(=O)OCC)(C(=O)NCCCN(C)C(C2CC2COC)=O)CCCCO1 Cc1nocc1C(=O)Nc1scnc1C(N)=O.C12C=CC(C1)C(=O)N2 N1(C(c2c(COC)cc[nH]2)=O)CCCCC12CC(NC(=O)CC1CCC(=O)N1C)C2 C=CC1(CC(=O)NCC(F)CNC(=O)C(CC(=C)C)NC(C)=O)CCCCC1 N1(Cc2cnc(CC)s2)CC2CCN(C(c3ccnc(Cl)c3)=O)C2C1 C(=O)(C1=CC(O)C(NC(=O)C(Cc2ccccc2)SCc2cccs2)C1)OC C1(NC(CCSCC)=O)C2CC3CC(C2)CC1(CNC(=O)COC(C)C)C3 c1(CCCC)ccc(C(=O)NCc2cccc(N3CCN(CC)CC3)c2)cc1N c1(OCCC(=O)NCC(N(C(C2C(=C)CC2)=O)C)C2CC2)c(C)cccc1C c1(OC)c(C(=O)NC2(CO)CCN(C(C3C=CCC3)=O)CC2)[nH]c2ccccc12 Cc1nc(NC(c2cccc(Br)c2)C(N)=O)[nH]c1C C#CC1CC2(CC2)CN1C(c1cc(CNC(c2c(C)cnn2C)=O)[nH]n1)=O CC1CCCn2c(C(=O)NCCCC3CCCN3C(=O)Cn3cccn3)cnc21 CCCC(C(O)C(=O)N(CC(C)(C)COC)C)NC(=O)CCCC(C)(C)C C(C)(C)(C(c1nnnn1C1COC1)NCCc1cc(CC)no1)OCC C=C(C)c1cccc(NC(=O)CC(CNC(C2COCCC2C)=O)OC)c1 C1(Cc2ccc(C)c(NC(CCCSC)=O)c2)CN(CC(O)C2CC2)CC(F)(F)C1 N1(C(CC2C(C)CCN(C(CC(C)N(C)C)=O)C2)=O)CC2CCCC(C1)N2C c1(CC(C)C)ccc2cc(C(=O)NNC(=O)Nc3c(Cl)cc(F)cc3Cl)[nH]c2c1 C12(NC(CC3C(C)CCCC3)=O)CCCC1N(C(c1cccc(F)c1)=O)CC2 c1(C(=O)NC2CC(C)(NC(c3c(O)cc(C)nn3)=O)C2)cnc2ccccn12 c1(-c2cc(C(=O)NC3C(NC(c4c(C)cco4)=O)CC3)no2)cccc(O)c1 CC(CN=c1[nH]c2ccc(N)cc2s1)NC(C1CN(C)CC(C)O1)=O CCC(C)(CCC(C)C)C(=O)N1CC(C(C)NC(=O)CCS(C)(=O)=O)C1 CCC(C)CC(=O)C(=O)NC1CCCCC1C(=O)NCC1(OC)CCCC1 C1(NC(c2c(CNC(CN3CCN(C)CC3)=O)n[nH]c2)=O)CCCCC1C#N C1(C(=O)Nc2scc(CCC(=O)OC(C)(C)C)n2)CCC(N)CC1 N1(C(C2CC(OCC)C2)=O)CC(F)(F)CC1CCNC(=O)CSc1nncs1 Cc1cc(CNC(C2CCN(C(C3CCC3(F)F)=O)CC2)=O)nnc1C N1(C(C=C(C)C)=O)CC2(CCC(CNC(=O)Cc3cn(C)nn3)O2)C1 N1(C(=O)CC2CN(c3cc(SC)ncn3)C2)CCCC(O)(C(N)=O)C1 C1(C(N2CCOC(CC(F)(F)F)C2)C(=O)NCCC(=O)OCC)CCSC1(C)C c1(C(=O)NCCC2CC(NC(C(C=C)(C)O)=O)C2)cc(Br)c([N+](=O)[O-])s1 Nc1cc(C(=O)NC2CCN(C(=O)CCn3ccnc3)CC2CO)ccc1Br c1(N2C(C)CC(NCc3ncccc3OCCO)C2)ncnc2cc(C3CC3)nn12 N1(C(C2(COCC)CCC2)=O)CCC(NC(=O)CCCCCSC)C2(CCC2)C1 C(C(CNC(c1cc(CNC(c2cnc(C(C)C)o2)=O)no1)=O)C(C)C)OC Cc1nc(Br)c(C(N2CC(C)(NC(C3C=CCC3)=O)C2)=O)s1 C1(C)(C(=O)NCC2(CN(C(c3c(Cl)cn(CC)n3)=O)C)CC2)CCCCNC1=O N1(CCCC(=O)NCC2N(C(CC3(C)CC3(Cl)Cl)=O)CC=C2)C(=O)CNC1=O N1(C(C(C)=C2CCCC2)=O)CCOC2CN(C(=O)C(C)OC(C)(C)C)CC12 c1(C(COC)(C)O)cn(CCNC(=O)C(Cc2ccccc2)SC)nn1 c1(C(=O)NC2(CC)CCN(C(C3SCCC3C)=O)CC2)cc(F)c(C)cc1Cl c1(CCNC(C(CN)N)=O)ccc2c(c1)OCCO2 CC1C(C(=O)N(CCCCN(C)C(C2CC2C(C)(C)O)=O)C)C1C C(=O)(C(F)(F)CCn1cc(-c2cccnn2)nn1)NC(=O)CCc1csc(Br)c1 c1(SC)nc(Cl)c(C)c(=NCC2CCCC2NC(C2CCc3cncn3C2)=O)[nH]1 C=C(Cl)CC(C(=O)N1CCC(CF)C1)NC(C1CC(=O)OC1(C)C)=O CC1(F)COCCN(C(c2ncoc2CNC(C2CC3C=CC2O3)=O)=O)C1 CCCCC(c1nnnn1Cc1ccccc1)NC(CCO)C1CC1 C#CC1CN(C(C2CCCC23CCC3)=O)CCN1C(=O)Cc1cc(C)n(C)n1 C(=O)(C1=CCCSC1)N1CCCC1.c12cc(ccn1)OC1CC(C1)CC(=O)N2 N1(C(CS(N)(=O)=O)=O)CCCC2(C1)CN(C(=O)C(O)CCC(F)(F)F)C2 CC1CCCc2ncc(C(N3CC(CNC(=O)CNC=O)CC34CCC4)=O)n21 N1(C(CCC=C)=O)CCCC(C(C)NC(=O)CCOc2ccc(C(N)=O)cc2)C1 CCC(CC(=O)N1CC(C)(OCC(=O)NCCC2CCOCC2)C1)C(F)F c1(C(=O)NC2CC(NC(C3CC3(F)Cl)=O)C(O)C2)ccc(CO)cc1F C1(NC(CSCCC)=O)CN(C(c2cc(C(C)(C)C)ccc2O)=O)C2(CCC2)C1 N1(C(COc2cccc(CC)c2)=O)CC(N(C(=O)Cc2cncs2)C)C(C)(C)C1 N1(C(C(C)CC2CCC2)=O)CCCN(C(=O)C2=NOCC2)C(CO)C1 N1(C(C(C)NC(=O)NC)=O)CCCC1Cn1cc(-c2n[nH]cc2C)nn1 c1(OCC=C)ccccc1C(=O)NCC1(F)CC(CNC(c2cnc(O)o2)=O)C1 Cc1[nH]nc(C(=O)NC2CC(CC(=O)NOC3CCC(O)C3O)C2(C)C)c1C CC(C)C(O)CC(=O)NC1(CO)CCCN(C(=O)Cc2cc(Cl)cs2)C1 C1(NC(c2ccc(OCCOC)nc2)=O)COC2(C1)CN(C(=O)CC(C)SC)C2 C(CCC(=O)NCc1cc(C(=O)NOC2CC2)co1)=CC c1(C(=O)NC2CC(C)N(C(=O)C=C3CCCC3)CC2)cnn2ccnc(N)c12 C1(C)(C(=O)NC(c2ncc[nH]2)C)CCCN(Cc2nc(-c3ccccc3)co2)C1 CC1CCC(c2nnnn2Cc2nnn(C)n2)(NC2CCCC2)C1 CC(N=c1[nH]c(=NC(C)CS(C)(=O)=O)c2sccc2[nH]1)C1CCOCC1 C1(C(=O)NCCN(C)CCO)COCCC1NC(=O)C=CC(F)F C=CCC(CNC(c1cc(O)n(CC)n1)=O)C(=O)NCC(C)SC C1(C(=O)NCCC2CC(NC(C(C)OC)=O)C2)C2COCC12 c1(C(=O)NC(CC)CNC(c2c[nH]ccc2=N)=O)cc2c(cn1)CCCC2 C1(CNC(CCC=CCC=C)=O)CCN(C(c2cc(Br)cs2)=O)CC1C CN(CCCC(=O)NCC1CC(O)CN1C(=O)C=CC1CCCO1)N=O C12(C(=O)NCC3(CC)CCOCC3)COCC1CN(C(=O)CCN(C)C)C2 C1(CCC(=O)NCC(CNC(C(CC)C)=O)(C)C)CCN(C)CC1 N1(C(C2C(NC(C(C)C(F)F)=O)CCO2)=O)Cc2ccccc2C1 CC(C)C(C(=O)NCCC1(O)CN(C(=O)CCC2CCCCC2)C1)C(C)C c1(C(=O)NCCCCNC(CNC(=O)OC)=O)cc(C)ccc1OC(F)(F)F C(=O)(C1c2ccccc2C2CC1C2)NCC(C1CC1)NC(CN(C1CC1)CC)=O Cc1ccc(C(N2CC(NC(=O)CC3CCC(=O)N3)C(N=[N+]=[N-])C2)=O)c(N)c1C Cc1ncc(CCC(=O)NC2CN(C(c3cc(C)[nH]c3C)=O)C2)c(O)n1 C(=O)(CC1CCCc2oc(C)nc21)NCC(C)(C1CC1)NC(C(C)=C1CC1)=O Cn1c(SCC(=O)NCC(C2CC2)NC(=O)C=CC=C(Cl)Cl)nc2ccccc12 n1(CCOC)cc(C(=O)NCCN2CCN(CCO)CC2)ccc1=O Cc1nnc2n1CCC2(C)C(=O)NC1CCN(C(=O)C(O)CC(F)(F)F)CC1 c1(C(=O)NC2CC(NC(C3C(C(C)(C)C)C3)=O)C2)cc(S(N)(=O)=O)ccc1O C1(NC(CSc2n(C)ccn2)=O)CN(C(c2cnncc2O)=O)CC1C1CC1 N1(C(C(C(C)C)C)=O)CCC2(CC1)C(NC(=O)C(C1CCCCC1)O)CS2(=O)=O c1(C(=O)NCC2CCN(C(C=C(CC)C)=O)C(C)C2)c(C)cc(Cl)cc1N c1(C(N(C)CC2N(C(c3c(C)cc(C)[nH]3)=O)CCC2)=O)cc(Br)c(C)nc1O N1(C(CC2CCC(C)CC2)=O)CC2(CCC(NC(C3CC34CCC4)=O)CC2)C1 Cc1nc(C2CCCO2)sc1C(=O)NC1CN(C(C23CC(F)(C2)C3)=O)CC1C N1(CC(=O)NC(c2ccccc2)C)CCCCC1C1CC1 c1(C(=O)NC2(C)CC(NC(=O)CC3CCCO3)C2)cc(Br)c2[nH]nnc2c1 Cc1onc(C(F)(F)F)c1C(=O)NC(C)CNC(C1CCCN1S(C)(=O)=O)=O C(C(C)C(=O)N1CCCC1C1CCN(C(=O)C(C)(C)OCC(F)(F)F)C1)OC N1(C(C(N2CCNC2=O)C)=O)CCC2(CCC2NC(=O)CC2(C)CCC2)CC1 CCCC(CC)C(=O)N1CC(F)CC1CN(C(=O)C(=O)N(C)C)C C(=O)(C1=CCOCC1)NC1C(NC(CC2C=NN(C)C2=O)=O)CCCC1 c1(OC)cnc(Cl)c(C(=O)NC2CCN(C(=O)CCC3CCCC3)CC2)c1 c1(C(=O)NC(CNC(c2cc(C)nn2C2CC2)=O)C)ccc2c(c1)OCCO2 C(CCNC(=O)Cc1cccnc1Cl)(C(C)C)NC(CN(S(CC)(=O)=O)CC)=O C(=O)(CCCCCCn1cc(CN)nn1)CC1CCCC(C(N(C)C)=O)C1 c1(-c2cc(F)c(CN3CC4CC3CS4=O)cc2)ccc2c(c1)CCO2 CCC(CC)CC(F)C(=O)N1CC(CC2CCCCO2)C1 C1(C(=O)NCC(CC2CN(C(C(C)C#N)=O)C2)(C)C)CCCN(CC(=O)N(C)C)C1 Cc1cccc(Br)c1C(C(=O)NCCOC1CCOC1)NC(=O)CC(O)C(C)C c1(C(=O)NCC(N(C)C(C23CC(C)(C2)C3)=O)C2CC2)cccc(C=C(F)F)c1 CP(C)(=O)c1cncc(C(=O)NC2CCC2CNC(C2CC23CCCC3)=O)c1 C(=O)(C#CC1CCCO1)NCCCN(C(=O)C(N1CCSCC1)C)CC c1(N2CCC(F)(C(=O)Nc3cccc(CCO)c3)C2)ncc2c(n1)CCC2 N1(CCCCCCCC)CCC2(CC1)CN(C(=O)C(C)NC(=O)CC)CC(C)O2 C1(C(=O)NC2(CCCC)CCC2)(NC(=O)COCCCC(C)C)CC1(C)C Cc1cc(NC(C2CCN(Cc3cccc4cccnc34)C2)=O)ncc1[N+](=O)[O-] C1(C(=O)NC)CCCC(CC2(CNC(COCCOC)=O)CC2)C1 c1(OC)c(C)cc(C(N2CC(CNC(=O)C#CC3CC3)N3CCC2C3)=O)cc1C C(=O)(C(C)(C)C(C)(C)C)NCCOCC(=O)NCc1nc(C(C)C)on1 c1(C(=O)NC2CCC(NC(CCC(=O)N(C)C)=O)C2)cnc(O)n(C2CC2)c1=O c1(CC(=O)NCC2CC2NC(C2(CO)CCOC2)=O)csc(-c2ccccn2)n1 c1(CC)ccc(C(=O)NCC2CC(NC(c3ccc(CO)o3)=O)C2)cc1F N1(CC=C)C(=O)NC(c2c(F)cnc(Cl)c2C)C(C(=O)OCC)=C1C1CCOC1 C1(C(N2CC(NC(c3ccc4nccn4c3)=O)(CO)C2)=O)CN=C2N=CNN2C1 N1(C(c2nc(OC)oc2)=O)CCCC2CN(C(=O)C(C)Cn3cccn3)CCC12 CCC(F)(F)CC(=O)NC1CCC1CNC(c1c(Cl)csc1Cl)=O CC1CCC(NC(C2CN3CCC2CC3)=O)CN1C(=O)CC1(O)COC(C)(C)C1 c1(CNC(c2[nH]ccc2CNC(C2CCCCC2F)=O)=O)c(F)cccc1F c1(C(C)N(C)C)ccccc1OC(c1cnc[nH]1)=O.C12CCC(C1)NC2=O c1(C(N(C(C)C)CCN(C)C(c2scnc2Cl)=O)=O)ccn2c1CSCC2 c1(C(C)C)nccc(=NCC(C2CCCCC2)CCO)[nH]1.C12CC1C(=O)NC2=O C(CNC(C1CC(O)C1)=O)(CCNC(=O)C(C)N1CC(C)C1)OC CC(C#N)CN=c1[nH]c2c(c(=NCCC3CC4(CCC4)CO3)[nH]1)CCCCCC2 c1(CNC(CCC=C)(C)c2nnnn2C(C)CC)cc2cnccc2o1 c1(C(N(C)CC2CCCN(C(C(C(=O)OC)C)=O)C2)=O)nc(O)nc(O)c1F N1(C(CC(C)(C)OC)=O)CCN(C(c2n[nH]cc2Cl)=O)C(C)CC1C c1(CC)cc2c(c(=O)o1)C(c1[nH]c(=N)sc1[N+](=O)[O-])NC(=O)N2CCF c1(C(=O)NCC(N2CC(CNC(CCNC(C)=O)=O)C2)=O)ccccc1C CC(C)C(C)CC(=O)NCCOCCCN(C)C(C1CCCC2(CC2)C1)=O c1(C(=O)NC2CCCC(NC(C(CC=C)CC)=O)C2)[nH]c2ccccc2c1CC C(CCCC(=O)NC1(CCCNC(c2cccc(C)n2)=O)CC1)SC CCCCCC(C(=O)NC)NC(c1csc(NCc2c(F)cc(Br)cc2F)n1)=O C(CC(O)C(=O)NCCCn1ccnn1)NC(=O)CC1CC(F)(F)C1 CC(C)(C)CC(O)CC(=O)NCc1cccc(-c2nn[nH]n2)c1 C#CCCN=C(NCC(CC)CC)NC(c1ccc(N2CCOCC2)cc1)C c1(C(=O)NCCCCCNC(CC(C)OC)=O)cc2ccc(Cl)cc2c(O)n1 c1(C(N(CC(C)(C)NC(=O)COCC2CCC2)C)=O)ccc(Br)cn1 C1(NC(C(C=C)O)=O)CCSC12CN(C(c1ccc(N(CCCC)C)cc1)=O)C2 CCS(=O)(=O)CC(=O)NCC(C)NC(C1CC(C)(C(=O)OC)C1)=O c1(C(=O)NCC(CNC(C2CCCN2c2cnccn2)=O)OC)sncc1C C1(C(=O)NC2CN(C(c3c(C)n(C4CC4)cc3)=O)CC2C)CCCNS1(=O)=O c1(NCC2CC(NC(C3(N(C)C)CCCCC3)=O)C2)ccc([N+](=O)[O-])cc1 c1(CCC)cc(O)ccc1CNCC(C)CC1CNC1 c1(OC)cc(OC)c(-c2nccn2-c2cccs2)cc1-c1nc(C(C)(C)C)no1 c1(C(=O)NC(C(C)NC(=O)CC2(CO)CC2)C)nccc2nn[nH]c12 N1(C(C2(C)CCCCC2)=O)CCC(CNC(=O)CCSC(F)(F)F)C(O)C1 N1(C(CC2(C(=C)F)CCC2)=O)C2CCC1C(C(=O)NCC1(F)CC(CO)C1)C2 N1(C(=O)NC(C#C)CC2CC2)CCCC1c1cc(C2CC2)on1 CC1(F)CN(C(=O)Cc2csnn2)CCN(C(c2c(F)ccc(F)c2Cl)=O)C1 CN=c1nc(N(C)CC2CCCN(C(C)C)C2)[nH]c(N2CCOC(C)(C)CC2)n1 C(=O)(C1=C(Cl)CCOC1)N1CCCC(NC(c2cnc(COC)s2)=O)CC1 N1(C(=O)COC2CCOC2)CCCC(C2CN(C(c3c[nH]c(C(F)F)c3)=O)C2)C1 CC(CC(C)NC(c1cc(C(F)F)on1)=O)NC(=O)CCOCC(F)F C(=O)(CCCC(=O)N(C)CCOCCC(=O)NCC1(C2CC2)CCC1)NCC Cc1cc(C)c(C(N2CC3CC3(CNC(=O)CC3(N4CCCC4)CC3)C2)=O)[nH]1 c1(CC)cccc(C(=O)NCC(C)(C)NC(c2cc(C(C)(C)C)oc2C)=O)c1N CC(C)C(O)C(=O)NCC1COCCN1C(=O)CCN1CCN(CCO)CC1 C1(C(=O)NC(c2c(OC)cccc2)CNC(=O)CCCF)CCc2ccccc2O1 c1(CC(=O)NCC2CCN(C(C=Cc3ncc(C)[nH]3)=O)C2)c(F)cccc1C#N C1(NC2CCN(C(COC)C)CC2)CC2CCC(C1)N2S(=O)(=O)C1CC1 c1(C(=O)NCCC(C)NC(c2ccccc2C2CC2)=O)cnn2c1CCC2 CC1CN(C(C2CC2C(=O)NCc2ccoc2C2CC2)=O)CCN1CCO C(CCN=C(NCC(F)F)NCC1CN(C)CCN1C)N1C(CC)CCCC1 Cc1cc(N)c(Br)cc1C(=O)NC(C)CN(C)C(c1cn(C)nn1)=O c1(CC)cncc(S(=O)(=O)NCc2ccc(C(F)F)nc2)c1 N1(C(c2nc(C)n(C(F)F)c2)=O)CCCN(C(C2CC2(Cl)Cl)=O)CC1C c1(C(=O)NCCN2CCN(C(C3CCC(F)C3)=O)CC2)cccc2[nH]nc(O)c12 N1(C(C(C(=O)OC)C)=O)CCC12CN(C(c1c(C)coc1C)=O)C2 c1(OC)cnc(Cl)cc1C(N1CCC(NC(C2(CO)CC(F)(F)C2)=O)C(F)C1)=O C1(C(=O)NCC2(OC)CN(C(=O)C(c3ccccc3F)C)C2)CCCC(C)CC1 c1(C(C(=O)NCC)N(C)Cc2ccn(C)n2)ccc(F)c(Br)c1 N1(C(c2cc(C#N)[nH]c2)=O)CC2(CCN(C(C34CCC(CC3(F)F)C4)=O)C2)C1 c1(C(N(CCOC)CCNC(=O)CCNC(C)=O)=O)ccc2c(c1)C(=O)OC2(C)C C(=O)(CCCCCCCC)NC(CC#C)C(=O)NCc1cncn1C CCCC(C)CN(C)CCN(C(=O)CCCC1CC1)C c1(C(N2CCCCC2CNC(C2(CO)CCC2)=O)=O)noc2ncccc12 c1(C(C(=O)N(CC(C)NC(C2(CC3CCC3)CC2)=O)CC)C)ccnn1C n1(COC)ccc(C(=O)NCC2CCC2NC(C2CCOC2C(C)C)=O)n1 N1(C(CCC(C)(C)OC)=O)CCC2CCCC12CNC(c1cccc(Cl)c1C)=O CC1(CCNC(c2csnn2)=O)CCN(C(C2(C3CC3)CC2)=O)C1 N1(C(CS(=O)(=O)NCC)=O)CC(NC(C2CC(F)(F)C2)=O)C2(CCC2)C1 C1(NCc2ccc(OCCC)cc2)CCCN(C(c2ncc[nH]2)=O)CC1 Cc1nn(C)c(C(c2nnnn2C(C)C)NCC(CO)C(C)C)c1Cl c1(C(N2CCC(N(C(=O)CC3CC(C(C)(C)C)C3)C)C2)=O)c[nH]nc1F N1(C(C(=O)NC(c2n(C(C)C)cnn2)C)=O)CCC(N2CCN(C)C2=O)CC1 CC1CC(C)N(C(=O)CCN(C(N)=O)CC)CCN1C(c1cc2c(ccn2C)[nH]1)=O c1(C(N2C(CNC(C(c3ccccc3)NC(C)=O)=O)CC2)=O)cc(Br)c(C#N)s1 c1(C(C(=O)N(C)Cc2cccnc2)NC(c2nnsc2N)=O)ccc(F)cc1 c1(C(N2CCN(C(CC(C)OC)=O)CC2CO)=O)ccc2nc(N(C)C)oc2c1 CC1CCCC(C)N(C(C23CC(NC(C4CCCCS4)=O)(C2)C3)=O)C1 c1(Cn2cc(CN3CC(C(=O)O)C(F)C3)nn2)ccc([N+](=O)[O-])cc1 C1(C(=O)Nc2c(Cl)nc(N(C)C)s2)CN(C(=O)COCC2CCOC2)C(C)(C)C1 c1(-c2cn(CC(N3CCN(CC(=O)NCC#C)CC3)=O)nn2)ccc(Cl)cc1F c1(C(=O)NC2CN(C(c3ccc(CC)cc3)=O)C2)cc2c(s1)CCS(=O)(=O)C2 N#Cc1ccc2c(=NC(=O)C3CN(Cc4cc(O)cc(F)c4)CCO3)[nH][nH]c2c1 C1(NC(c2c(OC)n[nH]c2)=O)(CNC(=O)C=CC(C)C)CCCCC1 n12c(-c3cnccn3)nnc1C2.c1ccc(COc2cccnc2)cc1 C1(O)(CN(C)C(c2cscn2)=O)CCCN(C(=O)CCOCC(F)F)C1 C1(C(N(CC(C)NC(=O)OC(C)(C)C)CC)=O)CCN1C(=O)CSC c1(C(=O)NCCCCNC(c2ccccc2)=O)cnccc1I N1(C(C)=O)CC2CCCC1C2c1nnc(CCCCOC(=O)N(C)C)o1 CC1=CCC(C)(C(N2CCN(C(=O)C=Cc3sccc3C)C(CCO)C2)=O)CC1 CC1COc2c(C(=O)OCC3CCc4cc(Br)ccc4O3)cnn2C1 N1(c2n(CCC(C)(C)SC)c(-c3cccnc3)nn2)CCOC(C2CCCO2)C1 C(=O)(C1=CC2CCCCCC12)N1CCC(C)C1CNC(c1ccc[nH]1)=O N1(C(c2c(C)[nH]c(=N)s2)=O)CCC2(CC1)CC2C(=O)NCCC1COC(C)(C)O1 N1(C(=O)C(F)F)CCC2C(C1)CN2C(c1cc(-c2ccccc2)nnc1O)=O C1(NCC(C(CC)CC)O)(NC(=O)OC(C)(C)C)CC2(CCCCC2)C1 O=C1CCCN(C(c2cc3cccn3cn2)=O)C(C(=O)O)C1 Cn1nccc1C(F)=CC(=O)NCC1COCCN(C(=O)Cc2cncs2)C1 Cc1c(NC(C2CC(CCNC(c3c(C)cccc3C)=O)C2)=O)cccc1CO C(C1CCCCC1)=CC(=O)NC1CC(CN(C)CC)C1.C1(=O)C(COC(C)C)N1 N1(C(C(C(C)(C)O)F)=O)CCCC(O)(CNC(=O)CCC(N)=O)CC1 C(=O)(C1=CSCCO1)NCC(C)NC(c1cc(-c2ccncc2)nn1C)=O c1(C(=O)NCc2cc(C(N(C(CCCC)C)C)=O)on2)cc(CC)oc1C C1(C(=O)NC(C)CNC(=O)OC(C)(C)C)CCC1S(N)(=O)=O c1(C(=O)NCC(CO)NC(C2CCN(C)C2)=O)cnc2[nH]nnc2c1 c1(C(N2C(C)C(NC(C34CC(O)C3C4)=O)CC2)=O)cccc2c1CCCC2 C(=O)(CC(C(F)(F)F)NC(=O)CCc1nc(C)no1)Nc1c(OC)ncnc1 c1(C(N2CCC(N(C(COCCCC)=O)CC)C2)=O)ccc(OC)cn1 Cc1cc(Cn2cc(C3(O)CN(C(=O)CN(C)S(N)(=O)=O)C3)nn2)n(C)n1 N1(C(=O)CC2CC=CCC2)CC2CCC1CN2C(=O)CC1CC2(CCC2)CO1 C1(NC(CCC#N)=O)CN(C(=O)CCOc2cc(Cl)cc(Cl)c2)CC12CC2 c1(C(N2CC(F)CC(C(=O)Nc3cc(F)cc(F)c3)C2)=O)ccnc([N+](=O)[O-])c1 C(C1=NOC2CN(C(=O)CC(F)(F)F)CC12)NC(c1ccc(COC)o1)=O C(N=c1nc(N(C)CC2COC(=O)N2)c2c([nH]1)CCS2)C1(OC)CCCC1 N1(C(c2cc(OC)no2)=O)CCC(C)(C)C1CNC(C1CCCN1C=O)=O Cn1c(O)ncc(C(N2CCCCC2CCCNC(=O)C2=CCCOC2)=O)c1=O c1(SC)nc(O)c(C(=O)NCC2CCN(C(=O)C(C)SC)C2(C)C)cc1C#N C1(NC(c2cc(CC)n(C)n2)=O)C2CCC1CN(C(c1ccc(Cl)c(I)c1)=O)C2 C(=O)(CC(C)(C)C#N)N(CCC(=O)NCC1(O)CC1)CC C(=O)(CCCCC(=O)c1ccc(NC(N)=O)cc1)NC(c1nc(=O)o[nH]1)C C1(C(=O)NC(CN(C(c2c(CC)cc[nH]2)=O)CC)C)CCCS(=O)(=O)C1 c1(OC)cc(C(=O)NC2CC2NC(=O)COc2cc(C)ccc2C)ccc1Br c1(C(Nc2ccccn2)=O)ccc(O)nc1.CC1CC1N(C)C=O C1(CC(=O)NCC2(NC(=O)CC3CC(=O)C3)CCC2)(OC)CCCC1 N1(CCCC)CCCCC1C(=O)NCC=CCNC(=O)C(O)C1CC1 CCC(C(=O)NCC(C)NC(c1nonc1N)=O)c1ccccc1 N1(C(C(C)OC)=O)CC2CC2(CNC(=O)CCc2ccc(OC(F)(F)F)nc2)C1 c1(C(=O)NCC(CNC(C2CC(S(C)(=O)=O)C2)=O)O)ccc(S(N)(=O)=O)c(F)c1 c1(N2CCC(C)C(NC(C3(C)CCC(F)(F)C3)=O)C2)ncccc1S(C)(=O)=O c1(C(N2C3C(C(=O)Nc4nnco4)C(C3)C2)C2(C3CC3)CC2)ccc(Cl)c(Cl)c1 N1(C(C2N(CCC(C)C)CCC2)=O)CCC(NC(c2ccsn2)=O)C12CC2 C1(C2CCOCC2)(CNC(CC(C=C)(C)C)=O)CCN(C(c2coc(O)n2)=O)C1 N1(C(C2(CC=C)CC2)=O)CCC(CNC(C2(C(C)(F)F)CCOCC2)=O)C(C)C1 c1(N(C(CNC(c2cnc(C)o2)=O)C)C)cc(C2CC2)nc(S(C)(=O)=O)n1 CC(C)C(CNC(=O)CC1CCCO1)C(=O)Nc1cncc(C2CC2)c1 O(NC(=O)CCN(C)C(C1CC(O)C(F)C1)=O)CCCOCC N1(C(C=CC(C)C)=O)C2CCC(C2)C1CNC(C1CCOC(C)(C)C1)=O O(N(C)C(=O)CN=c1[nH]c2c(c(=NCCC3CCOC(C)C3)[nH]1)CCCC2)CC C(CCCCC(=O)NOCCCO)NC(C1(OCC)CCCC1)=O N1(C(C2CCC(C)(CC)O2)=O)CCC(C2CC2)C1CNC(=O)CN1CC2CC2C1 C=C1CCN(C(=O)C=CCCC(C)C)C(C(=O)NCCNC(=O)CO)C1 N1(C(c2n(CC=C)ccc2)=O)CCC(CNC(=O)C(C)OCC(F)(F)F)C12CC2 C1(NC(C(C=C=C)C)=O)CN(C(=O)CNC(C2CCC2)=O)C2CCCCC12 C1(C(N(C(C)CC2CC2)C)=O)COCCN(C(C23CCC(C)(C2)OC3)=O)C1 Cn1c(C(=O)NC2(CCNC(=O)CCC3CCCC(=O)N3)CCC2)cnc1Cl Cc1ccsc1C(=O)NCc1nocc1CC(=O)NOCCCN(C)C C1(NC(=O)C=CC=C(Cl)Cl)CCCC12CN(C(=O)C=CCOC1CCOCC1)C2 c1(C(=O)NC2C(C)CN(C(C3C4CNC(=O)C34)=O)C2)cc2ccncc2s1 Cc1cccc(C)c1C(O)C(N1CCC(F)(CNC(c2nc(C)n(C)n2)=O)C1)=O C(=O)(CC(O)C(Cl)(Cl)Cl)NC(COC)CNC(c1ccc(N(C)C)cc1)=O C1(CC(N2C(CC(C)(C)C)CC2)=O)CC(C)(C)CN1C(C1CC(=O)C1(C)C)=O N1(C(CC=CC=C)=O)CCN(C(=O)C(O)C2CC2)CC1CO C1(NC(C2CC(=C)C2)=O)COCCN(C(c2[nH]cnc2C)=O)C1 C1(CCOC)(NC(=O)CCC2CCCN2C)CCN(C(C2CCCN2C)=O)CC1 CC1(CNC(c2ccccc2C2CCC2)=O)CCN(C(=O)CC2(O)CCOC2)C1 C1(CC)C(NC(c2cccc(F)c2C)=O)CCCN1C(=O)CNC(N)=O c1(OC)cc(F)c(F)cc1C(=O)NC1C=CCN(C(=O)COc2ccon2)C1 c1(OC)cccc(OCC(=O)N(C2CCN(C(c3cc(Cl)cn3C)=O)CC2)C)c1 N1(C2(C(N(CCN(C(C3C(C)C3C)=O)CC)CC)=O)CC2C(F)(F)F)CCOCC1 CC(=Cn1ccnn1)C(=O)N1CCC12CN(C(c1cc3cccnc3[nH]1)=O)C2 c1(C(=O)NCC2CN(C(c3c(CC)ncnc3)=O)C2)cn2cc(Cl)cc(Cl)c2n1 C1(CCC)CN(C(c2ccncc2CC)=O)CC1NC(c1ncc(F)cn1)=O c1(C(=O)Nc2ccc(C#C)cc2Cl)cnc2c(Br)c[nH]c2c1 N1(C(C(=O)NCCOc2cccc(OCC)c2)=O)CCOC2COCC2C1 c1(OC)cc(N2CC(CNC(=O)C=CCO)CC2C)nc(C(F)(F)F)n1 Cc1cc(-c2cn(CCCN(C)C(C3(C)CC3(F)F)=O)nn2)ccc1Br CCC(C)(C(=O)NC(CCN(C(=O)CN(C)C(C)C)C)C(C)C)C(F)F c1(CCC)c(C(=O)NCC2CCCCC2NC(=O)C(C)SC(F)(F)F)nnn1C Cc1cccc(Cl)c1NC(=O)COC1CCOC1.N12CCC(C)(C1)CC2=O CC1CCCC1(c1nnnn1C1COC1)NC1(C)CC1 c1(C(=O)NCC(=O)NCCC(=O)NCCC2C(C)C2)ccc(C#N)n1C c1(C(=O)NCC2N(C(c3c(CC)nc[nH]3)=O)CC(O)C2)c(C)ccc(OC)c1N N1(C(C2(C=C)CCN(C(C3SCCS3)=O)C2)=O)CC2OC(=O)N(C)C2C1 C(=O)(CC(C1CCCC1)NC(=O)C(N1CCC(Nc2ccccn2)C1)=O)OC c1(-c2c(C)cc(C(=O)NCCCCN(C)C)nc2)cccc2c1CN(C)C2=O N1(C(CCCCCC=C)=O)C(CNC(=O)CCc2ccsc2)CC2CCCCC12 C1(C2(O)CN(C(=O)C(=O)NCc3c(OC)ccc(Cl)c3F)C2)(C(=O)OC)CCC1 CC1=CCSC1C(=O)NC(C)CCCNC(C1CCC1C#N)=O C1(CCNC(C2(C)CN(C(CCC)=O)C2)=O)CCOC(C)C1 CCC(C)CCC(=O)NC1CN(C(=O)CN(C2CCSC2)C)CC1(C)C CC(CN(C)C)CC(=O)N1CCC(C(=O)N(CC(C)(O)C2CC2)C)CC1 C(=O)(CCC(C)(C)O)NC1C(OC)CN(C(=O)CN2CCCCC2)C1 C#CCCCCCNC(C1CCC(NC(c2c[nH]c(=NC)o2)=O)C1)=O C(=O)(CC(C(F)F)NC(=O)C1=CCSC1)NCC1(C(C(C)C)O)CC1 C(CCCCC(=O)N(C1CCCN(C(C2CCCCC2(F)F)=O)CC1)C)N(C)C c1(C(C(=O)NC2C(NC(C3C(CC)CCO3)=O)CC2)(F)F)ccc(C)cc1 c1(OC)cccc(C2(C(N3CCOC(CNC(C4CCSC4)=O)C3)=O)CC2)n1 c1(OC)cc(C(N2C3CN(C(=O)CCc4cccc(O)n4)CC23)=O)cc(Br)c1 CCC(CC)CCCN(C(=O)CCNC(=O)CC(C)=C(C)C)C Cc1cc(P(C)(C)=O)oc1C(N1c2ccccc2C(C)C1C)=O C1(F)(COC(C(C2CCCCCC2)C)=O)CCCCC1 C1(C(=O)NCCCC(C)NC(C=CC(C)(C)SC)=O)CCc2c(ncn2C)C1 CC1CC(NC(=O)C(=O)NC2CC2)CN(C(=O)CCCCc2ccc(F)cc2)C1 c1(C(=O)NC(CC)CN(C)C(C2CC2c2ccsc2)=O)nc(O)c(C)s1 N1(C(=O)OCC)CCCCC(c2n(-c3c(NC(C)=O)cccc3C)nnn2)CC1 Cc1ccc(Br)c(F)c1C(=O)NCC1(O)CCCN(Cc2ccc(O)cc2Br)C1 C1(C(N2C3CN(C(CCc4cnn(C)n4)=O)C(C3)C2)=O)Cc2cccnc2C1 c1(C(N2CCN(C(C3CC4(CC(=C)C4)C3)=O)C(C)C2)=O)ccn2c(O)nnc2c1 C1(NC(C(C)=C(CC)C)=O)CC2CN(C(C3(C(F)F)CCCO3)=O)CC12 CCS(=O)(=O)CCCCCN1CCCC1CNC(C1CNC(=O)CC12CCC2)=O C(=O)(C(C(C)(C)C)N1CCCC1=O)N(C(CNC(c1c(CC)cno1)=O)C)C c1(CCNC(C2CCN2C(c2ccc(F)cc2O)=O)=O)ccc([N+](=O)[O-])cc1 CCCCC(C(=O)N1CCCC(F)C1)NC(c1ccc(Cl)s1)=O c1(C(=O)NCCCN(C(=O)C(O)CC2CC2)CCO)cc2c(cn1)OCCC2 c1(C(N2CCC(C)(NC(C(C)C(C)(F)F)=O)C2)=O)cnn2c1C(=O)NCC2 Cc1cc(C(=O)NCC(C)CC(=O)NC(C)Cc2cnccn2)nnc1O c1(OC)cc(C(=O)NCCN(C)C(C2CC2CF)=O)c(F)cc1N c12ccsc1NC2=O.C1(C(N2CC(OCCNS(C)(=O)=O)C2)=O)CC=CCC1 C(c1cnccc1C)=CC(=O)NCC(CC=C)NC(=O)C#CC1CC1 CC(C)(CNC(C1CCCC(NC(=O)CCC2CCC2)CC1)=O)CC(F)F C(=O)(CCCCC(N)=O)NCC1N(C(COC2(C)CCC2)=O)C2CCC1C2 c1(Oc2ccc(NC(C3(C)CCCN3)=O)cn2)cc(Cl)ccc1C(F)(F)F C1(NC(c2cc(C(C)C)[nH]n2)=O)CN(C(c2nccnc2Cl)=O)CC1O c1(C(N2CCC(C(=O)NC3(C)CCCC3C)(CC)C2)=O)ncnc(O)c1F C(CN=c1nc(N2CCc3nc(Br)sc3C2)c2c([nH]1)CSC2)OCC(F)(F)F N1(C(COC(CC)C)=O)CCC(C(C)(C)C)(CNC(=O)Cc2sc(C)cc2C)C1 O=C(CN=c1ccc(Cl)n[nH]1)NC1CCCC12CN(C(=O)CC1CC3(CC3)C1)C2 C1(NC(c2c(C)n(C)nn2)=O)C2CC3CN(C(c4cc[nH]n4)=O)C1C3C2 N1(CC(=O)NCC2OCC(CNC(C(C)(Cl)Cl)=O)C2)CSCCSC1 CCC(C)CCC(=O)NCCNC(=O)Cn1cc(C(F)(F)F)ccc1=O N1(C(C2C(CNC(c3c(C)nccc3)=O)C2)=O)CC2(COC(=O)N2C)C1 N1(C(C(=O)NC)CC2CCC(C)(C)CC2)CCc2cncnc2C1 [N-]=[N+]=Nc1ccc(NC(C2(NC(=O)CC3CC(=O)C3)CCOCC2)=O)cc1 C1(COC)CN(C(=O)CCC(C)(C)N(C)C)CCN1C(=O)C1CC1 c1(NCc2c(Cl)cn(C)n2)ccc(S(=O)(=O)NCCc2cncs2)cc1Br C=CC(CC)CC(=O)N(C)CC1CN(C(=O)CC2OCCCO2)CCO1 N1(C(CCN2C(=O)CCC2)=O)CCCN(C(=O)COC2CC=CC2)CC1CO C(CC(C)(C)C(=O)NC1CN(C(c2ccc(CO)c(F)c2)=O)CCC1C)OC C1(C(CNC(c2c(OC)n[nH]c2)=O)(C)O)CCCN(C(=O)OC(C)(C)C)C1 C1(CNC(C(COC)(C)OC)=O)CCCC2(CN(C(c3ncccc3F)=O)C2)O1 C(=O)(CCC(C)(C)C)N1CCCC(CN(C)C(c2ncc(Cl)nc2Cl)=O)C1 c1(OC)noc(C)c1C(=O)NCC(N1CCN(C(=O)C(C)=C(C)C)CC1)C Cc1ccc(C(CC2CC2(C)C)OCC(=O)NC2CC(F)(F)C2)cc1F C1(C(=O)NCC(CC)NC(C2(C(=O)OC)CC2)=O)CCC(SC)C1 CCC(CNC(c1cc(C(N)=O)c[nH]1)=O)N=c1[nH]c(Cl)ncc1[N+](=O)[O-] N1(CC(N2CCC3CN(C(C4CC4F)=O)CC32)=O)C(=O)Cc2ccccc2C1=O c1(C(=O)NC2C(CNC(C(C)SC)=O)C2)ccc2c(c1)CCN2S(C)(=O)=O n1(CCNC(c2n(CC=C)nnn2)(C)CC2CC2)c(O)nc2ccccc12 c1(C(N2CCC2(C)CC)C(=O)NCC(=C)C)cnc(Br)s1 N1(C(C(N2CCOC2=O)C)=O)C2CCCC1CN(C(=O)CCc1cnoc1)C2 c1(C(N(CC(C)(C)NC(=O)C#CC2CCC2)C)=O)cccc2ncccc12 N1(C(C(CCC)OCC)=O)CCN(C(c2nc(O)sc2C)=O)CCC1C CC(C(=O)NC1CC(CNC(c2cnn(C3CCOC3)n2)=O)C1)C(F)F N1(C(CSCC(N)=O)=O)CCN(C(=O)CC2CCN(CC(F)(F)F)C2)CC(O)C1 C12(C(N(C)CC3CCC(F)C3)=O)CC(CO)(CN1C(=O)C#CC1CC1)C2 C1(C(=O)NC2(CNC(C=C3CCC(C)C3)=O)CCCC2)CCc2ncsc2C1 N=c1cc(C(N2CCOCC2CNC(C2(CO)CC2)=O)=O)cc[nH]1 Cc1ccc(OCCC(=O)NCC2CCCC2NC(c2c[nH]nc2F)=O)c(C)c1 CC1(C)CC(NC(C2CCC3(CC3)N2C(=O)C(F)OC(F)(F)F)=O)C(=O)O1 c1(CNC(c2n(CCCC)nnn2)C2(C)CCCS2)ccccc1C1CC1 C=CC(C)(O)CC(=O)NCC1CCC12CN(C(=O)CN(S(=O)(=O)CC)C)C2 S(=O)(=O)(c1ccc([N+](=O)[O-])cc1F)C(c1ccn2cncc2c1)C(=O)O N1(C(C(c2cccc(Cl)c2)(C)C)=O)CCN(C(=O)C=CC2CCCO2)CC(O)C1 C(=O)(CCN=c1[nH]ccs1)N1CC2=C(CN(C(C34CCC(OC)C3C4)=O)C2)C1 C1(NC(CCN(C)CC)=O)(CC)CCCN(C(C2C3CC4C(C3=O)C24)=O)C1 C1(NC(C(c2ccccc2F)C)=O)CN(C(=O)CCNC(=O)CO)CC1O Cc1csc(C(=O)NC2COCC2CNC(=O)CCCc2cccnc2)c1 Cc1nc(C(C)C)ncc1C(=O)NC1(C(C)(C)C)CCN(C(=O)CCC(N)=O)C1 C1(C(=O)NC2CC(CC)(CC)C2)CN(C(C2CCO2)=O)CCN1C CC1(C)CCCC(CNC(c2nc(Cl)c(Cl)s2)=O)CC1 N#Cc1cc(C(N2CCCC2C2CCN(C(c3nc(Br)c[nH]3)=O)C2)=O)cs1 c1(C(=O)OC)ccc2nc(CNC(N3CCC(CO)C(F)C3)=O)[nH]c2c1 C1(C(=O)NC2C(NC(c3c(C)con3)=O)CCCC2)CN(CP(C)(C)=O)C1 S(=O)(=O)(c1cnc(NCC(C)C(F)F)c(Cl)c1)NCC1(CC)CCOC1 N1(C(CC(C)F)=O)CCC(F)(CNC(=O)C(c2cccc(Cl)c2)(C)C)CC1 c1(C(N2CCC(NC(C3CCC(C)O3)=O)C2C)=O)cc(O)nc2ccc(F)cc12 CC(C)C(O)C(=O)N1CC(CNC(c2cn(CC3CNC(=O)O3)nn2)=O)C1 N1(C(CS(CC(C)C)(=O)=O)=O)CCCCC2(CCN(CC3CCC3)C2)C1 n1(CC(=O)NCCNC(C2C(C)(C)S(=O)(=O)CC2)=O)ncn2cccc2c1=O CC1CCC(=CC(=O)Nc2nc(Cc3cccs3)cs2)C1 C1(C(N2CCCCCC2)=O)CC(F)(F)CN1C(=O)CC1CCCSC1 CS(=O)(=O)C1(N2CCN(C(C3CCC4CNCCN34)=O)CC2)CCCCC1 O=C(CCCc1cccnc1)OCCC1CSC1 C1(CC)CN(C(=O)COCC2CC2)CCC1NC(=O)C1CC1 C1(C(N2CC(OCCNC(c3c[nH]nc3C(F)F)=O)C2)=O)CS(=O)(=O)C1 c1(C(N(CCCCCNC(COCC(=C)C)=O)C)=O)c(C(F)(F)F)n[nH]c1C Cc1nc(=N)[nH]cc1C(=O)N(C)CC1CCCN(C(=O)CCCCC2CC2)C1 N#Cc1cc(=NCc2nnc3ccccn23)c2cc(Br)ccc2[nH]1 C1CC(C(C)C)O1.C(C(C(=O)N1CCC1CC(N)=O)n1cc(CC)nn1)OCC C(CC1=CCN(C(c2ccccc2-n2ccnn2)=O)CC1)NC(C12CCC1C2)=O C1(CNC(C(CC2CC2)OC)=O)CCN(C(c2ccc(O)cc2F)=O)CC1(F)F Cc1ccc(Cl)c(C(N2CC(NC(c3cnc(C(F)F)s3)=O)C3CC23)=O)c1 N1(C(c2c(CC)n[nH]c2)=O)CCC(C)(CNC(c2cc(C(F)(F)F)on2)=O)C1 N1(C(CN2CC(C)(OC)C2)=O)CCC(NC(c2cnncc2C)=O)C1C(C)(C)C Cc1cnc(C(=O)NC2(CCC(=O)NCC(O)CC3CCC3)CCC2)cn1 c1(NC2CCCC(NC(CN(CCCCCC)C)=O)C2)ncc2ncnc-2[nH]1 CC(C)CCC(F)C(=O)N1CCOC(C(=O)N(C)Cc2cnccn2)C1 C(C)(C)(CCCNC(=O)CC1CC=CC1)NC(C(C)N(C(C)=O)C)=O C(c1ccsc1)=CC(=O)NCC1COCC1NC(=O)CSC1CCCCO1 c1(-c2cncc(C(C3CCNCC3)C)n2)c(F)ccc(C)c1F.c12nc(ncc1F)NC2C C1(NC(C(=O)NCC(=O)N(C2CCNC2)C)=O)C2CC3CC(C2)CC1C3 Cc1ccc(C(N2CC3CC2C3C(N2CCCC(C)C2CO)=O)=O)c(I)c1 c1(C(N2CCC(N(C(=O)C=Cc3cnn(C)c3)C)C2)=O)ccc(C(F)F)cc1Cl N1(C(C(C)(C)OC)=O)CCN(C(=O)CC2C(=O)ON=C2C)C(C2CC2)C1 c1(C(C)NC(c2n(C(C)C)nnn2)c2nncn2C)ccc(Cl)cc1 C1(C(=O)Nc2cnccc2CCO)CCCC(NC(C2(F)CCCCC2)=O)CC1 C#CCCCC(=O)NCC(CC)NC(=O)C(C(C)C)Nc1ccccc1 C1(NC(c2n(CC)ccc2)=O)CCN(C(c2cc(CCO)on2)=O)CCC1(F)F C12(NCC(=O)NCC3N(C(=O)OC(C)(C)C)C(=O)CC3)CCCC1OCC2 c1(NCCF)ncnc2c1ncn2CCc1c(F)cccc1Br C1(NC(CN(C)S(N)(=O)=O)=O)CN(C(=O)CC2(C)CCCCC2)CC12CCCC2 C1(C(=O)OC(C)C(N2CCN(c3ccccn3)CC2)=O)CCC2C(C1)C2(F)F CCCC(C#N)C(=O)NCC(C)C(N1CCC(C#N)CC1)=O Cc1cc(CCC(N2CCCC(C(C)NC(=O)CN(C)C)C2)=O)ccc1Cl N1(C(c2c(Cl)cn(CC)n2)=O)CCC2C(C1)CN2C(=O)C(C)c1ccco1 Cc1cccc(CN(C(=O)CC(O)CNC(=O)C(C)C2CC2)C)n1 N1(C(C(CC)C)=O)CC2CCCN(C(C3C(c4ccccc4)C3C)=O)C2C1 C(CNc1c(C2(C(=O)O)CC2)cccc1)(C(C)C(C)C)OC c1(NC(N2CC(F)CC(C(=O)Nc3ccc(C)cc3)C2)=O)c[nH]c2ncccc12 c1(C(N2CCN(C(CCC#C)=O)CC2CC2CC2)=O)cnc2nc(O)ccc2c1 CC(C)(C)CC(F)C(=O)NC1CC=CCC1C(=O)NC(CO)C(N)=O c1(CC)ncc(Br)cc1C(=O)N(C1CCN(C(=O)C(F)C2CC2)CC1)C CCC(C)C(O)C(=O)NCCCCNC(c1cnoc1C)=O c1(-c2nc(-c3ccc(SC)cc3)nn2CC2CCCCO2)cc(Cl)c(C)cn1 C(=O)(C(C)(C)C(C)(F)F)NC1CCCC(NC(c2cc(OC)c(O)cc2)=O)C1 C=CCCCC(C(=O)NC1(C)CC(F)(F)C1)NC(=O)CCNC(N)=O c1(CNC2(c3nnnn3C)CCCC(N(C)C)C2)noc2cc(F)c(F)cc12 N1(C(c2cc(OC)no2)=O)CCCC1(C)CCC(N1CCC(C)(F)C1)=O N1(S(C)(=O)=O)CCc2ccc(C(=O)NCC3(Br)CC3(F)F)cc2C1 N1(C(c2cc(CC)on2)=O)CCOCC(F)(CNC(c2ccc(OC)s2)=O)C1 N1(C(C2C(CCC)C2)=O)CCC2(CC1)CN(C(c1nsc(OCC)n1)=O)C2 C1(C(=O)NCCCCC)CCN(C(=O)CCC(N)=O)C(C)C1 CC(CC(=O)NCC1CCC(NC(=O)C(C)(O)C(F)(F)F)C1)C(F)(F)F C1(NC(CCC(=C)C)=O)CC2CCC1N2C(=O)C1=CCOCC1 c1(C(N2CCOCC(CNC(CSCC)=O)C2)=O)cc(F)cc(F)c1F N1(C(C(CC2CN(C(=O)COC3CC3)C2)F)=O)CCC(F)(F)C(F)C1 C1(NC(=O)CC2(N(C)C(C3(CC)CCCCC3)=O)CC2)CC2(C1)CC21CC1 N1(C(CC2CCCC(C)(C)C2)=O)CCC(CNC(c2cnco2)=O)C(F)(F)C1 Cc1sc(C(c2nnnn2C(C)(C)C)NC(C)CCC(C)C)c(Br)c1C C=CC(C)(O)CC(=O)NC1CC2(C1)CC2NC(C1C2(CC2)C12CC2)=O C1(CN(C(c2ccsc2SC)=O)CC)CCCN1C(=O)CCc1ncc(C)[nH]1 Cn1cc(NC(C2(CNC(=O)CC34CCCC3C4)CC3(CC3)C2)=O)c(Cl)n1 C(=O)(C1=CCCSC1)N1CC(SC)C(NC(=O)CNC(c2ccncc2)=O)C1 c1(NC(=O)OC(C)(C)C)ccnc(OC(C2COCC23CCC3)=O)c1 N1(C(C2OCCC(=O)C2)=O)CCCCCCC1C(=O)NCC1CC12CCC2 c1(C(=O)NCC(C)(O)CNC(c2cc(F)cc(Cl)c2N)=O)ccc([N+](=O)[O-])cn1 c1(C(CC(C2(NC(C(C3CC3)OC)=O)CC2)OC)=O)nc(OC(C)C)ccc1Cl Cc1cc(=O)c(C(N2CCOC(CNC(c3sc(F)cc3C)=O)C2)=O)c[nH]1 C1(C(=O)NC(C)CCc2cn[nH]c2)CCN(C(=O)C(C)N2CCCC2)CCO1 c1(C(=O)N(c2cccs2)CC=CCNC(C2C(C(=O)OC)C2)=O)cn(CC(N)=O)nn1 C=CC1(CNC(=O)C(C)CNC(=O)CCC2CCOC2)CCOCC1 C1(NC(CCCC2C(C)C2)=O)CCCC(NC(c2cn(C)nc2Br)=O)CC1 c1(C(=O)NC2CC3(CC(NC(C4(C)CCOC4)=O)C3)C2)ccc2c(c1)CCOC2 C1(C(N(C2CCN(C(c3cnc(OC)s3)=O)C2)C)=O)Cc2cccc(F)c2O1 CC1(C)CCC(C(N2CCC(NC(C3CC3[N+](=O)[O-])=O)C2(C)C)=O)CC1 C=CCCCCCCC(=O)N1CCCCC1CN(C)C(C1CC1C(N)=O)=O c1(C(N2CC(C)(CC(=O)Nc3ncc(F)cn3)C2)=O)ccc2[nH][nH]c(=N)c2c1 C1(NC(=O)Cc2ccc(O)cn2)C2CCC1CN(C(=O)CCC1CCCOC1)C2 C1(CNC(c2csnc2Cl)=O)CCCN(C(=O)C(F)n2cccn2)CC1 N1(Cc2nc(N(CCCO)C(c3ccccc3)C)c(Cl)[nH]2)CCCC(O)(n2ccnn2)CC1 C1(C(N2CC(C)N(C(=O)CC3OCCO3)CCC2)=O)CCc2ccccc2C1 C1(C)(Cn2cc(CN(C)Cc3nn(C)nc3C(F)(F)F)nn2)CCCC1O C(CC(CC)C(=O)NCC1CC(F)CN1C(=O)Cn1ncc(Cl)c1C)=CC c1(CC(C(N2CCC(CN(C(=O)C=CCO)C)C2)=O)O)ccc(Cl)cc1 C=C(Cl)CCC(=O)NC(Cc1cc[nH]n1)C(=O)NC(c1ccncc1F)C C1(OC)CC(CNC(C2CC(O)C2)=O)N(C(=O)CCn2ccccc2=O)C1 N1(C(CCC=CC)=O)CCC(NC(c2n[nH]c3cc(C)ccc23)=O)C2(CCC2)C1 C(=O)(CC1CCOc2ccccc21)NCCN(C(C(CC(=C)C)OC)=O)CC c1(NC(=O)NC(c2cnsc2)C)ccccc1OCC=CCN c1(CC(=O)NC2CCCC(NC(CC(CN(C)C)O)=O)C2)nc2c([nH]1)CCCC2 N(C(=NCC(C)(C)OC(F)F)NCC1CCCO1)C1C(C(C)(F)F)C1 c1(C(N2CCC(N(C(C3CCS3(=O)=O)=O)CC)C2)=O)cc2n(c1)CCSC2 N1(C(c2c(C)[nH]cc2)=O)CC(C(=O)NC2CCOCC2C)C(C)C1 C(C(C(=O)NCC1CCC=CCC1)C(C)(C)C)NC(C1C(C)CC(=O)CC1)=O CCCC(C)(O)C(=O)NC1CN(C(=O)CS(=O)CC)CC1CC1CC1 c1(N2CCC(NC(=O)Cn3ccc([N+](=O)[O-])n3)C(F)C2)ncc([N+](=O)[O-])cc1Br C1(N(C(COCCOCC)=O)C)CCCCC1NC(c1cc(C)on1)=O c1(CC(N2CC(O)(C(C)NC(c3ncccc3F)=O)C2)=O)cccc(O)c1F N1(C(=O)Cc2cc[nH]c2)CCCC(CC(N2CCCC(c3nc[nH]n3)C2)=O)C1 C=CC(C)CC(=O)N1CCC(C(=O)NC2CC2CC)(OC)C1 C1(C(C(=O)NCC=CC)C)CN(C(c2cc(=O)cc[nH]2)=O)CCO1 C1(CNC(CC(C)c2ccco2)=O)CN(C(c2cc(Cl)cn2C)=O)CC(C)(C)C1 C1(NC(Cc2c(OC)cccc2)=O)CC1C1CCN(C(c2cn[nH]c2)=O)CC1 N1(C(=O)CCCc2cccs2)CCC2(CCN(C(C3CC4C=CC3C4)=O)C2)C1 N(C(=NCCC(C)=O)NCc1cc(C)ccc1O)CC(C(=O)OC)OC N1(C(CN(C)S(N)(=O)=O)=O)CCCC2(C1)CN(C(c1cscc1C(F)F)=O)C2 C(C)(C)(C(C)NC(=O)C(C)=CC1CC1)NC(C(C)OCCSC)=O c1(C(C)C)ccccc1NC(N1CC2CC1C2C(=O)NC(C)C(F)(F)F)=O c1(Nc2onc(CC(CCC)N)n2)ncnc2ccsc12 C1(NC(c2cccc(C(C)(F)F)n2)=O)CC2CN(c3nnc(O)s3)CC2C1 c1(C(=O)NC(CCC)C2CCCC2)ccc(CNC(C2CCC2C#N)=O)nc1 C1(CNC(c2n(C(CC)C)ncc2)=O)CN(C(=O)CSCCOC)CC(C)(C)C1 CCCCC(CC)C(=O)N1CCN(C(C2CC(OCC)C2)=O)CC1COC C1(O)(CCNC(CCOCCN(C)C)=O)CCN(C(=O)CCC2CC2)CC1 S(=O)(=O)(c1ccc(NC(CN2CCCC2)CO)cc1Br)NC(CC=C)CO c1(C(N2CCC(CCCNC(c3nc(C)oc3)=O)CC2)=O)ccc(C#N)c(O)c1 C1(C(C(=O)NCC(CO)NC(CCC)=O)O)CCCCCC1 c1(C(N2CCCC(N(C(C=CSC)=O)CCF)C2)=O)cc(NS(C)=O)ccc1F N1(C(C(CC)C)=O)CCC(C)(C)C1CNC(=O)C(=Cc1ccncc1)C Cc1cnc(C(=O)NCCC2CCC(NC(=O)CCC3CCCOC3)C2)c(F)c1 Cc1cccc(C(N2CCOCC2C(=O)NC2CCC(F)(F)CC2)=O)c1O C1(CCNC(c2n(C)ncn2)=O)CCCCN1C(=O)CCc1ncc[nH]1 C1(CNC(c2c(C)nc(CN3CCNCC3)o2)=O)CCCC2(CCC2)C1O c1(OC)cnccc1C(=O)NC1CCC(F)(CNC(C2(OC)CCCCC2)=O)C1 Cc1ccn2cc(C(=O)NCC=CCNc3cc(C)c([N+](=O)[O-])cn3)nc2c1 c1(C(N(CCCCNC(C(c2cnn(C)c2)OC)=O)C)=O)nn[nH]c1C(F)(F)F C1(C(=O)NCCOCCCNC(C2(C)CSC2)=O)CCCC(C2CC2)O1 c1(CC)ccc(NC(C2CC(C)CN2C(c2cc(C)[nH]n2)=O)=O)c(C)n1 C1(C(N(CC=C)CCC)=O)CC(C)N1C(=O)CCNC(=O)CO N1(C(C=Cc2n(CC)ncc2)=O)CCC(CNC(C2(F)CC=CC2)=O)C(F)(F)C1 c1(C(=O)NC(CNC(C2(C)CC2)=O)C2CCC2)c(F)c(N)cc(Cl)c1F C1(C(=O)NCCc2ccn(Cc3ccccc3)n2)CC(=O)N(Cn2cccn2)C1 Cc1cccnc1CC(=O)N(C)CC1CCCN1C(=O)CCSc1ccccc1 c1(CN(C)CCNC(=O)C(=O)NCc2ccc(F)cc2)ccc(Br)cn1 C(=O)(C(N(CC(C1CCCS1)=O)Cc1cccs1)C1CC1)NCCC C1(C(=O)NC2CCCC(NC(c3nc(C)sc3)=O)C2)CNC(=O)CC1(C)C C=CCC(C)(CC)C(=O)N1CCC(C=CC(=O)NC(C(N)=O)C2CC2)CC1 n1(C(C)C)cnc(C(=O)NC2CC2NC(=O)Cc2ccsc2Cl)c1 N1(C(C=Cc2scc(C)n2)=O)CC2(CCN(C(c3cc(N)ccc3C)=O)C2)C1 C(=O)(C(C)(C)CC#N)NC(C1CCCN(C(C(C)=C2CCCC2)=O)C1)C C(CCN(C)CC)(C(C)C)NC(=O)NC(COC(C)C)C(C(=O)C(C)C(C)C)=O CC1CN(c2nsc(CC(F)(F)F)n2)CCS1(=O)=O c1(-c2nc(CCC)nn2Cc2cccc(F)c2)cc2ncc(Br)cn2n1 N1(C(C2=C(C)OCCS2)=O)CCCC2CN(C(=O)CCC3CCCC3)CCC12 CCC(C)CCC(O)CC(=O)N(c1nc(C(C)C)cc(C)n1)C.C12CN(C1)C2=O CC1CCC(N(C)CCNC(c2nnnn2C)Cc2cc(C#N)cs2)(CO)C1 c1(OC)ncccc1CC(=O)NCC(C1CCN(C(=O)C=CC2CC2)CC1)C c1(OCc2nc(C(C)C)on2)ccc2c(c1)CCC2.N12CCC(C1)N(C)C2=O c1(C(=O)NCC2CN(C(C(CSC)O)=O)C(C)(C)C2)ccc2c(c1)CCS2(=O)=O O=C1CN(CCNC(C2CCC(NC(c3ccc(Cl)cn3)=O)CC2)=O)CCN1 C(=O)(N=c1nc[nH]s1)C1N(Cc2ncc(C)nc2)C2C(C1)C2 S(=O)(=O)(c1ccccc1Cl)NC1CN(Cc2c(C)ccc(O)c2)CC1C#N N1(C(C2CC(C(=O)NCc3cncs3)C2)=O)CCC(O)(c2ccccn2)CC1 CCC1=C(C(=O)NCCN2CCN(C(=O)C(C3CCCO3)OC)CC2)SCCO1 C#CCCCCC(=O)N(CC(O)CNC(=O)CCc1ccc(CC(C)C)cc1)C c1(C(C)C)ccc(C(c2nnnn2C2CC2)NCCc2cnc(C(C)O)s2)cc1 c1(C(=O)NC2CC(N(C(=O)CC3CC3(C)C)C)C2)c[nH]cc1Br c1(OC)ccc(C2(C(=O)OCCCCc3nc(C)cs3)CCC2)cc1 N1(C(CC2CCC(=O)NC2)=O)CC2(CC2)CC1C(=O)NCCOCCCF Cc1ccc(C(=O)NCC(C2CCCC2)NC(=O)CCCN=[N+]=[N-])c(N)c1C N1(C(c2c(CC)scc2)=O)CCCC(C(C)N)C1 CC1(C)CCCC(C(N2CCC3(CC2)CC3CNC(c2cnc(S)[nH]2)=O)=O)CC1 C1(C(N2CC(COC)N(C(=O)C=CC(=O)N(C)C)CC2)=O)CN2CCC1(C)CC2 Cc1cc(C(=O)NCC2CC(F)CN2C(c2ccc(C)nc2)=O)cc(O)n1 N1(CC(=O)NCC(CC)NC(C(C)(C)OCCC)=O)CCCCC1=O c1(C(=O)NC2C(CNC(=O)CN3C(=O)CNC3=O)CCCC2)ccn(O)c(=O)c1 N1(C(=O)CC(O)C2CC2)CCC(F)(CNC(C2(O)CC2)=O)CC1 N1(c2nc(C)nc(Cl)c2)CCCC(C2CCN(C(=O)C=C3CCC(C)C3)CC2)C1 N1(C(C2C(C)(C)OC2(C)C)=O)CC2CC(C1)CN(C(C1CCCO1)=O)C2 N1(C(c2c(C)nn(C)c2C)=O)CCc2[nH]nc(-c3ccsc3)c2C1 O=C(C#CC1CCCC1)NCC(O)C(=O)NC1CC(CCF)C1 c1(C(=O)NC(C)CCNC(=O)C(C2CCCCC2)O)cc2cccnc2nc1O c1(C(=O)NC2(C#N)CC2)cccc(-n2cc(C3CCC3)nn2)c1.N12CCC(CC1)C2 C(C1CN(C(=O)C(C)C(=O)OC)CC1C(=O)NCCC1CCC(=O)N1)=CC Cc1ccc(F)cc1C(=O)NC1C2CC1N(C(=O)Cc1nnc(S)n1C)C2 Cc1ncn(C)c1C(=O)N(CCNC(=O)C(C)C(C)C)C1CC1 c1(N2CCC(N3CCN(C(CCC)=O)CC3)C2)nc2c(OCC)ccc(Br)c2s1 C1(CNC(C2N(C=O)CCC2)=O)CN(C(c2ccc(O)nn2)=O)CC12CC2 c1(C(N2CCC(CNC(C3N(CCC)CCC3)=O)C2)=O)cc(C)cc(Cl)n1 CC1COc2c(C(=O)NC3CCC(CNC(c4cc(Br)c[nH]4)=O)C3)cccc21 N1(C(c2cc(OC)c(F)cc2)=O)CCCCC2(CCN(C(C34CC3C4)=O)C2)C1 CC(C)CC(O)C(C)C(=O)NCCC(O)C(=O)NCCCc1ccccc1 c1(OC(C(=O)N(C(CNC(CCC#C)=O)C)C)C)cccc(Br)c1 N1(Cc2c(-c3cccc(OC)n3)cccc2)CCCOCC12CC2 C1(C(N2C(C(N3CC(CSC)C3)=O)COCC2)=O)CC2(C1)CC2(F)F C1(C(N(C2CCCN(C(=O)CCc3cn[nH]c3)CC2)C)=O)CC2(C1)CC(C)(C)C2 N1(C(C)C(=O)NC2CC(CCNC(=O)CCC3CC3(F)F)C2)CCOCC1=O C(C(C)(C)C(=O)N1CCN(C2CCCN(C(=O)Cc3ccc(Cl)s3)C2)CC1)SC C1(C(=O)NC2(CC#C)CCC2)CCC(C)(C)N(C(=O)CCC2CC2)C1 N1(C(COC2(C#C)COC2)=O)CC2CC(NC(c3cc(C(C)C)no3)=O)CC2C1 c1(C(=O)NCCCNC(c2cc(C)nn2C)=O)cc2ccc(C)n2cn1 C1(CC(N2CC(C)C(NC(=O)C(N3CCC(O)CC3)C)C2)=O)CN2CCN1CC2 c1(NC2CCCS(=O)(=O)CC2)ncc2ccccc2c1C(F)(F)F c1(CC(N2C(CC(=O)NCC(=O)NC)CCC2)=O)c[nH]c2cc(F)ccc12 N1(C(C)C(=O)N(C)C)CC2(CCC(C(=O)NC3CCN(CC4CC4)CC3)O2)C1 C(CCCCCF)NC(C(Cc1cn[nH]c1)NC(C(CC1CC1)OC)=O)=O N1(C(C(CSC)C)=O)CC(NC(c2cc(N)ccc2O)=O)CC12CCC2 CCCCC(CN=c1[nH]cncc1Br)NC(=O)CCNC(C1(c2cccs2)CC1)=O c1(OC)cc(C)c(NC(C2(C)CC(NC(=O)CC3CCOC3(C)C)C2)=O)cn1 c1(C(=O)NC2CC(C)(NC(C(N3CCCC(O)C3)C)=O)C2)ccc(O)c(O)c1 CC(C)(C)CC(O)CC(=O)NCC1CC2(CCC2)CN1C(=O)COC(=O)CO c1(C(=O)NCC(C)(C)Nc2snc(CCOC)n2)cc2sccc2cn1 c1(C(=O)OC)ccnc(NC(c2cccc(Cl)c2)Cc2cccc(C)c2)n1 C(N=c1cc[nH]cc1C#N)C1(F)CCN(C(C(C=C)(C)CC)=O)CC1 c1(C(=O)NC2CN(C(CN(C3CC3)CC)=O)C3C2C3)cc2ncccc2s1 C1(CNC(C2C(=O)NCC2)=O)CN(C(C2CC3(CSC3)C2)=O)C2(CCC2)C1 C1(C)(CNC(c2cnc(SC)s2)=O)CCCN(C(=O)CC2CCCCC(=O)N2)C1 C(=O)(CCC(=O)NN(C)C)NC1CCN(C(C(CN(C)C)(C)C)=O)CC1(C)C C1(CC(=O)OC)CC(CNC(=O)CC2CC(NC(C3CC3(C)C(F)F)=O)C2)C1 C(C(C)(C)CNC(C1C=CCC1)=O)N(C(=O)CC1CCCC1O)CC c1(C(N2CCCC(OC3CC3)C2)C(=O)NC(CC)(C)C)cncc(C(C)(C)C)c1 N1(C(C(CC#C)(C)CC)=O)CCC2(C=C(C(=O)NC(C)COCC3CC3)C2)C1 N1(C(c2c(CC)con2)=O)CCCC2CN(C(=O)CN3CCS(=O)CC3)CCC12 C(=O)(CC(O)CC(C)(C)C)N1CCC(C(N(CC(CC)O)C)=O)(CF)C1 c1(C(=O)NCC2C(NC(c3ncn(C)n3)=O)COC2)ccc(Br)cc1C#N C1(C(N2CC(OC)C(NC(c3n[nH]c(C)c3F)=O)C2)=O)COc2ccccc2C1 C1(CN(C(C(C)OCC#C)=O)C2CC2)CCCN1C(c1cnn(C(F)F)c1)=O CS(=O)(=O)CCC(=O)N1CCCCC(C(=O)NCCCc2ccccn2)C1 C(C(=O)NC1CCCN(C(c2nocc2Cl)=O)C1)(C(C)(C)C)SC N1(C(C)=O)CCCC(C(N2CCCC(Nc3ncc(O)cn3)C2)=O)C1 N1(C(C(C=CC)O)=O)CC(C(=O)NCc2cccc(C)n2)C(CC)C1 CCC(CNC(c1ccccc1)C1(O)CCC1)CC(F)(F)F c1(C(=O)NCC(C)(C2CC2)NC(C(C=CC)O)=O)cnc(F)c(F)c1 CN1C(=O)C(CC(=O)N2CC3CN(C(C4(O)CC4)=O)CC3(C)C2)c2ccccc21 c1(OC)ccc(CC(=O)NC2CCCC2CNC(=O)CCNS(C)(=O)=O)cn1 C(C1CCCc2cccnc21)NC(=O)CC(C(F)(F)F)n1cccn1 c1(N2CC3C(NC(=O)CSc4ccncc4)(CCC3)C2)ncnc2cnccc12 C=CCC(C)(C)C(=O)N1CC(O)(CNC(=O)CCSCCCC)C1 C1(NC(C2CCCC(C(=O)OC)C2)=O)CC2CCC1CN(C(c1ccoc1)=O)C2 CC1CN(C(=O)C(C)(C2CC2)N(C(=O)Cn2ccnc2)C)CCCO1 CN=c1[nH]cc(C(N2CC(CO)(NC(C3CC3C(F)(F)F)=O)C2)=O)s1 N1(CC(C)C)CC(C(=O)NCC(C)CN(C)C(c2cc(C(F)F)on2)=O)CC1=O CN1CC(NC(=O)C(CN=[N+]=[N-])NC(C2CCCC23CCC3)=O)C(F)(F)C1 Cc1cc(C(=O)NC(C)(CNC(c2cc(C(N)=O)co2)=O)CO)nc(O)n1 C#CC1(C(=O)NCCC(C)C(F)F)CN(C(c2nscc2C)=O)C1 C1(CNC(C(CC)OCC)=O)C(CC)CCN1C(=O)CC(C)(C)C1CC1 c1(C(=O)NCC(C(C)C)NC(C(C=C)O)=O)cnc(C(F)(F)F)c(C)c1 c1(NCC(C(C)C)(C)C)ccc(S(=O)(=O)NCC2(CCO)CCOC2)cc1F C1(COC)(CNC(=O)CCc2ccsc2)CCN(C(=O)C(C)(C)CN(C)C)CC1 CC#CCC(CO)NC(C1CCCCN1C(C12CCC(C1)C2)=O)=O Cc1ccc(CC(=O)NC2(CC3CC3)CCN(C(C3C4CN(C)CC34)=O)C2)cc1 C(=O)(CC(O)c1ccccc1)N1CC(CN(C(C2(CC=C)CC2)=O)C)C1 c1(CC(=O)NC23CCCN(C(C(CC)O)=O)C2C3)csc2nc(C)cn12 C1(C(=O)NCCC2N(C(C3(C)CCN(C(C)=O)C3)=O)CCC2)CCCCCCC1 Cc1cc(F)c(CN2CCC(C(C)C(=O)Nc3cncc(F)c3I)CC2)c(Br)c1 C1(C(N(C)CCc2cnn(C)c2)=O)CCC2(CC2)N1C(C1C2CCCOC12)=O c1(C(=O)NCCCN(C(=O)Cc2nnc(O)s2)C(C)C)cc2nnn(C)c2s1 c1(C(=O)NCCCC(C)NC(=O)CCC2CC2(F)F)cc(C(C)C)nc(Cl)c1 c1(C(N(CC(C)(C)NC(=O)CCP(C)(C)=O)C)=O)nn(C)c2c1CS(=O)(=O)CC2 CC(C)(C#N)C(=O)NCC1CCN(C(=O)Cc2ccnn2C2CCC2)C1 c1(N2CC(O)CC(C)C2)nccc(=NCc2ccc(-n3cccn3)cc2)[nH]1 N1(C(C2(C#C)CC2)=O)C2CCC1(CNC(=O)CSCCOC)CC2 CCCCC(CC)CC(C(=O)NCc1cccc(Br)c1)N1CCC(C#N)C1 CCC(CC(=O)NC1CCC(N(C(=O)CNC(N)=O)CC)CC1)C1CC1 C1(CCNC(=O)CO)(OC)CN(C(=O)CCNC(=O)CN(C)C(C)C)C1 N1(C(C2C(C)C2)=O)CCC2(CC1)CN(C(=O)COCc1ncnn1C)CCO2 C(CC(C)(C)C(=O)NCc1ocnc1C(=O)Nc1ccc(F)c(O)c1)SC N1(C(c2nc(CCC)oc2)=O)CC2CC(NC(C3CCCC3(C)C)=O)C1C2 C1(NC(c2cc(C(=O)OCC)nn2C)=O)CCCCCN(C(=O)C(C)CF)C1 O=C1CC(C(=O)NCCC(N2CCC2OCCOCCOCC2CCC2)=O)=NN1 c1(N(C(=O)C(C(=O)OC(C)(C)C)C2CCC2)C)ccc2c(c1)CC(=O)N2C c1(CCC(N2CCCCC(NC(C3C(=O)NCC3)=O)C2)=O)cc2ccccc2[nH]1 C1(CC)CN(C(=O)C(F)C(C)C)CCC1CNC(C1CCCC(=O)N1)=O N1(C(CCCN(C(C)=O)C)=O)CCC(C(=O)N(c2ccccc2C)C)C(C)(C)C1 CC(c1cccs1)=CC(=O)NC(C)C(C)(C)NC(c1cc(C2CC2)ns1)=O c1(N(C2CC3(C2)CC(N)C3)Cc2cnc(OC)c(Br)c2)ncnc2ccsc12 c1(CC(N2C(CCNC(C3(OC)CC3)=O)COCC2)=O)ccc2c(c1)CC(C)O2 Cc1[nH]nc(Cl)c1NC(C1CCN1Cc1cnc(Cl)cn1)=O C1(C(=O)NCC(CC)NC(=O)CCCCCF)CC12CCC(F)(F)CC2 CCCCCC(O)C(=O)N1CCN(C(c2c(CC)nn(C)c2CC)=O)CCC1C S(=O)(=O)(c1cc(C(=O)NCC2(C)CCC(NC(=O)C(C)=CC3CC3)C2)co1)NC c1(CC)ccc(C(=O)NCC2CCCCN2C(=O)CCN2CCCC2)cc1F N1(C(C2N(C(C)=O)CSC2)=O)CC2CCCC(NC(c3scnc3Cl)=O)C2C1 c1(NC2CCN(C(Cc3ccc(C)cc3)=O)C2)cc(C)nc(CO)n1 CC1CN(C)CC(NC(=O)C(N2CC3CC2CN3CCCC(C)(C)C)=O)O1 C1(C(N(C2CCCN(C(c3ccc(C(F)F)s3)=O)CC2)C)=O)CCC2CC1CO2 N1(C(C(CCSC)NC(C)=O)=O)CCN(C(=O)CCCC2CCC2)CC(CO)C1 C1(N(C(CCCN(C(C)C)C)=O)C)CC2CC1N(C(c1cncc(N)n1)=O)C2 N1(C(C(C)n2ccnn2)=O)CCOCC1C(=O)N(C1CCN(C)C1=O)C C(=O)(C(F)CCC(C)(C)C)NC1CCC(C(=O)NC2CCC(C(=O)OC)C2)CC1 n1(CCC=C)c(N2CCC(C(C)(C)C)(C(=O)OCC)C2)nnc1C1CC(O)C1 c1(CN(C(c2cc(Cl)ccc2Br)=O)CCO)cccc2cc[nH]c12 c1(C(=O)NCCn2cc(CNC(c3n(C)ccc3)=O)nn2)ccccc1CO S(=O)(=O)(c1ccc(N2CCN(CC(C)(F)F)CC2)cc1Br)NC(C)CC#N Cc1nc2[nH]c(C(=O)NCC3CCC3NC(c3ccccc3)=O)cc2s1 Cc1cc(C)c(CC(N2CCC(NC(=O)CC3CC4CC4C3)C2C)=O)s1 CCCC(CC)CCC(=O)NCC(C(N1CC2CCCC(O)C2C1)=O)C(C)C c1(C(=O)NC2C(NC(CCC(=O)NC)=O)COCC2)ccc2nsnc2c1 Cn1nc(I)cc1NC(=O)NCC1CC(n2cccn2)C1 Cc1ccc(C)c(CN=c2ccc(-c3cnn(CC#N)c3)c[nH]2)c1O CC(C)C(CNC(c1occc1C1CC1)=O)NC(=O)COCC(F)(F)F.C12CC1C2 CC1CN(C(C2(CNC(=O)Cc3ccnc(O)c3)CC=CC2)=O)CC1(F)F C1(C(=O)NC(C2CC=CCC2)C(=O)N(CCC)C)CC(=O)NC(=O)N1 c1(C(C)NC(=O)NCC2CC2(C)C)cccn1C c1(C(N(CC(O)CNC(=O)CS(N)(=O)=O)C)=O)ccc(=NCC2CC2)[nH]c1 N1(C(c2c(C)nc(CNC(C3CCN(C)C3=O)=O)o2)=O)CC(C)(C)CCC1C c1(NC(CC)CSC)cc(S(=O)(=O)N2CCCOC2)ccc1C#N C1(CC(N2CC(O)(CNC(c3cc(C4CC4)no3)=O)C2)=O)CCCC(C2CC2)O1 C(CN=C(NCC1CCC(F)(F)CC1)NC1CCCC(C(N)=O)C1)OCC=C CC#CCC(C(=O)N1CCC1CF)NC(c1c[nH]nc1CC)=O c1(CN2C(C(=O)Nc3c(C(C)=O)cccn3)CC2)c(Br)cccc1Br S(=O)(=O)(C(C)CN=c1[nH]c(N2CCn3c(O)nnc3C2)nc2ccsc12)NC N1(C(=O)NC2CCCC23CCC3)CCCN(c2ccccc2)CC1 c1(C(N(C(C(=O)NC2CN(C(CC)=O)C2)C)CC)=O)cc2cnccc2[nH]1 C1(CC(=O)N(C)CCN(C)C(c2ccnn2CC(F)(F)F)=O)CCCC(C)(C)O1 C1(CC(=O)N(CCN(C(C=CC)=O)C(C)C)C)CCCN(C)C1 N1(C(C(C)C#N)=O)CC(C(=O)NCCN(C(C)C)C2CC2)CC(C)C1 c1(C(=O)NCCN(C)C(C2C3COCC23)=O)cccc2cccnc12 C1(CNC(CC=CC=C)=O)CC2(CCN(C(c3ccc(C(N)=O)cc3)=O)C2)CO1 c1(C(=O)NCCC(C)NC(C23CC=CCN2CCC3)=O)ccc2c(c1)CCC2 C(=O)(C(C)C(C)C)NCC(C)(CNC(c1sc(C)nc1C)=O)OC N1(C(C(CC)n2nccc2C)=O)CCN(C(c2cn(C3CC3)cn2)=O)CC1CO C(CC(=O)NCC(O)CNC(=O)C(C)c1ncco1)NC(=O)OCC c1(C(=O)NC2COCC2CNC(c2ccncc2F)=O)cc2cc(Cl)ccn2n1 c1(CC)ncc(C(=O)NC(C)CC(C)NC(c2c(Cl)sc(C)c2C)=O)c(C)n1 C1(CNC(C2C(OCC)C2C)=O)CCN(C(=O)CC2(OC)CC2)CC1 C(=O)(CCCc1ccsc1)NC1CC(NC(CC)=O)C1 C(CC(F)F)(C(=O)N1CC2(CCC2O)C1)NC(=O)C(C1CC1)C1CC1 C1(CNC(CSc2n(C)cnn2)=O)CN(C(=O)CCSCC(N)=O)CC1O C(C(=O)N(C)CC1CCN(C(=O)CCc2ncc[nH]2)C1)(C(C)C)NC(=O)OC CC(C)CCCCCC(=O)N1CC(NC(=O)C(C)OC2CCCCC2)C(F)C1 c1(C(=O)NCC2C(NC(C3(C)CC=CCC3)=O)CCC2)cc[nH]c(=N)c1[N+](=O)[O-] Cc1ccc(C(=O)N(CCNC(c2cn(C)nc2Br)=O)C(C)C)nc1C c1(C(=O)NCCCN(C(C2CC2C#N)=O)CC)nccn2c(Br)cnc12 c1(C(=O)NC2CC(F)(CNC(CNC(CC)=O)=O)C2)cc(C#N)ccc1Cl N1(CC(=O)NC(CC=C)CNC(c2csc(-c3ncc[nH]3)n2)=O)CCCNC1=O c1(C(=O)NCC(C2CCN(C(C3COCCO3)=O)CC2)F)ccc2nc[nH]c2c1 c1(CN2C(C)(C(=O)OCC)CC2)nc(OC)cc(C)n1 CCCCC(F)(F)C(=O)N1CCC(c2cn(Cc3cc(C4CC4)no3)nn2)C1 C(CC(=O)N(C)CCc1cc[nH]n1)(CC(C)C)NC(c1c(OC)scc1)=O CCCC(C#N)C(=O)N(C)CC1CCCCN1C(c1ncc(F)cc1F)=O c1(C(=O)NCC2(C)N(C(c3c(C)c(Cl)ccc3)=O)CCC2)cc2c(ccn2C)[nH]1 C1(COC)C=CCCN1C(C1COCC1NC(=O)CC(C)SC)=O c1(C(=O)NC2CC(O)CN(C(c3ccnn3C3CC3)=O)C2)cccc2sccc12 c1(C2(NC(c3nnnn3C)C)CC2)c[nH]nc1C.c12nnnn1C2C1CC1 CC(C)C(C(=O)N(C)CC1(C#N)CC1)C(C)NC(=O)COc1ccsn1 CC(CC#N)C(=O)NC1CCN(CCCNC(=O)CS(C)(=O)=O)C1 C1(NC(=O)C=CCN2CCCC2)CCCC(NC(=O)Cc2cc(CO)on2)CC1 C(C)(CC(=O)NNC(=O)C(C)(C)CCCCNC(=O)CC1CCCOC1)OC C12(CN(c3nccs3)CC(C)C)CC(c3ccccc3)(C1)C2(F)F c1(N(CC(C)C#N)C2CC2)ncnc2c1ncn2C1CC1 N1(C(C2N(C(CCC=C)=O)CC(N=[N+]=[N-])C2)=O)CC2(CCC2)OCC1C c1(-n2c(C(c3c(C)nc(Br)s3)NC3CCSCC3)nnn2)ccc(F)c(Cl)c1 C(CN=c1[nH]c(=NC(C)CC(N)=O)[nH]c2cc[nH]c12)C1CCN(C(C)C)CC1 CCC(CC)CCCNC(=O)CN(C(c1cnc(C)cc1C)=O)CC1CC1 C1(CNC(c2cncc(O)c2)=O)CCCCN1C(=O)Cn1ncccc1=O c1(NC(CCC)CCCNC(=O)C(F)CC2CC2)nccc(C(N)=O)c1[N+](=O)[O-] CC1(C)CC(NC(c2cccc(C3CC3)c2)=O)CN1C(=O)CC1CCCOC1 c1(OC)nc(Cl)ccc1C(N1CCCCC(NC(C2(O)CCCCC2)=O)C1)=O Cc1ccccc1CC(C)Nc1cc(N(C)CC2CC2)ncn1 c1(CN(C)CC)c(-c2ccc(OCc3cncn3C)nc2)ccnc1OC c1(NCc2cnc(C)[nH]c2=N)nc[nH]c(=NCC2CC(F)(F)CO2)c1C C#CCCC(O)C(=O)NC1CCN(C(=O)C(C)(C)CSC)C1 N1(C(Cc2cncc(C)c2)=O)CC(NC(=O)C(F)C2CCOC2)CC2(CCC2)C1 CN(C)NC(=O)CCC(=O)N1CC2C(NC(c3cccc4oc(O)nc34)=O)C2C1 C1(NC(Cc2cc(C)no2)=O)CC2CC1CN(C(=O)COC(C)C)C2 C1(NC(C=Cc2cc(C)no2)=O)C2CCCN(C(=O)C=CCN(C)C)C2C1(C)C N1(C(C2CCCC2(F)F)=O)CC23CCCC2(C1)CN(C(C1C2COCC12)=O)C3 Cc1cc(C(=O)NCCC(C)(C)NC(=O)CS(C)(=O)=O)c2cnn(C(C)C)c2n1 c1(CC)ccc(C)cc1NC(C1(CNC(=O)CC2(C#N)CC2)CC12CCC2)=O N1(C(CCC(C)NC(C2(CC(=O)OCC)CC2)=O)=O)CCCN(C(C)C)CC1 C1(C(=O)NC(c2nc[nH]n2)CC)C2CC(O)C(C2)N1C(=O)CS(=O)(=O)CC N1(C(c2c(=N)cc[nH]c2)=O)CC2CC1CCC2NC(=O)CCCS(N)(=O)=O c1(C(=O)NC(c2ccccc2)CC=C)cc(C)cc(I)c1O N1(C(c2cn(CCC)nn2)=O)CC(CNC(=O)C(=O)NC2CC2)C(F)(F)C1 C1(NC(c2cnn(C(C)C)c2F)=O)CC(NC(C2(C)COC2)=O)C12CCC2 C1(F)(C(N(CCOCCNC(c2nc(CCCC)sc2)=O)C)=O)CCS(=O)(=O)C1 C(=O)(CC1=CCCC1)NCCC(=C)CNC(c1cc(F)c[nH]1)=O CC1(C)COCC1CC(N1CCC(NC(=O)C=C2CCC2)C1)=O c1(CCC(=O)NCC(C)(O)CNC(c2ccnnc2O)=O)ccccc1[N+](=O)[O-] C1(NC(CSC(C)C)=O)CC2CCC(C1)N2C(c1ccc2c(c1)COC2)=O c1(CNC(C2CN(S(=O)(=O)CC3(C)CCOCC3)C2)C)ccc(Cl)c2ccccc12 CC1Cc2c[nH]nc2C(C(=O)N2CC3CCC2C(NC(=O)CN(C)C)C3)C1 Cc1ccc(NC(=O)C(=O)NCCC2(NC(c3csnc3Cl)=O)CC2)cc1 Cc1nn2cc(C(=O)NC(C)(CNC(=O)C(C(C)(C)C)N(C)C)CO)nc2s1 Cc1ccc(C=CC(N2CC(NC(c3cccc(F)c3F)=O)CC(O)C2)=O)cc1 CC(C)C(C)CNC(=O)CCN(C(=O)Cn1nccn1)C1CC1 N1(CC2(C(=O)NCc3ccc(Cl)c(Br)c3F)CCC2)CC2CCCCC2C1 C12(NC(c3nc(C)nn3C)=O)CCCC1N(C(=O)Cc1cnns1)CCC2 C(=O)(C1CCc2cccc(F)c21)NCCCC(C)NC(=O)CN(C)C(N)=O CON1CC(C(=O)NC2(C3CCCN3C(c3ncccn3)=O)CC2)CC1=O C(=O)(C(C#N)C(C)(C)C)NC1CCC(C(N2CCC(C(C)C)CC2)=O)CC1 C1(O)(CNC(C=C(COC)C)=O)CCN(C(=O)C(c2cccc(O)c2)C)CC1 C1(OC)CC(CNC(c2ccc(Br)s2)=O)N(C(=O)CNC(C)=O)C1 N1(C(C2(CC=C)CCCC2)=O)CCCC(C2CCN(C(=O)C(O)CCC)CC2)C1 N1(C(c2sc(C)c(C)c2C)=O)CC(C)N(C(c2cn(C)ccc2=O)=O)CC1C N1(C(CC(CC)C)=O)CCN(C(=O)C(C)(C)OC(C)=O)CC1CCOC C1(CNC(C=CCOC)=O)(COC)CCCN1C(=O)Cc1ccc(Cl)cc1 C1(c2nn[nH]n2)(C(=O)NC2CC=C(C)CC2)CCN(CC2C(C)=NNC2=O)CC1C N1(C(c2n(C(C)C)ccc2)=O)CCC2(CC1)CC2C(=O)NC1CCC2CCC12 CC(C)CC(CCO)N=c1nc(N2CC3C4CCC(C4)C3C2)c2c([nH]1)CCCC2 C(=O)(C(C)(C)C(O)C(C)C)N1CCCC(CN(C(c2cc(OC)ncc2)=O)C)C1 C=C(Cl)CC(C(=O)NCc1csc(C)c1)NC(C1CC(=O)CS1)=O Cc1cc(C(=O)N(C)CC2CCCN(C(=O)CCC3CC3(C)C)C2)c(F)cc1Cl C(=O)(C1=C(Cl)CCCC1)NC1CCN(C(c2ncc(OC)cn2)=O)CC1F C1(NC(C2(C)CC(C)OCC2)=O)CCC(N=c2ccnc(Cl)[nH]2)CC1 C1(NC(c2cccc(C)n2)=O)CCN(C(=O)CN2CC3CC3C2)C(C)C1 C(N=c1[nH]c2cccc(Br)c2o1)C1CCN(C(c2cc(OC)ns2)=O)C1 N1(C(Cc2cn(CCCCNC=O)nn2)=O)CCNCC(O)C1 N1(C(C2CN(c3ccn(C)n3)C2)=O)CC=CC(C(=O)NCC(O)C(F)F)C1 Cc1cc(=NC(CNC(C2(C)CC2Br)=O)C2CCC2)nc(-c2cccs2)[nH]1 C1(NC(C(CC)(C)O)=O)CC2CCC1CN2C(=O)C(C)Cc1cnc[nH]1 C(C)(CCN(C)C(C1CC(C(=O)OC(C)(C)C)C1)=O)NC(CN(C(C)=O)C)=O N1(C(COCCCOC)=O)CCC(C(F)(F)F)C(NC(c2cn(C)cc2C)=O)C1 C=CCCC(CC(C)C)C(=O)Nc1cccc(NC(=O)Cn2nnnc2C)c1 Cc1cc2ncc(C(=O)NCC34CC3CN(C(=O)CC3(CO)CC3)C4)c(C)n2n1 c1(CC(=O)NC2(CC)CCCN(C(C3C(=C)C3)=O)C2)c[nH]c2c(F)cccc12 C1(Cl)(C(=O)NC2C(CNC(C(N3CCCCC3=O)C)=O)CCC2)CC12CCC2 CN1C(=O)COCC1CNCC1CC2CCCC2C1 C1(NC(=O)CC2CCCC2O)CN(C(c2cc(Cl)nc(Cl)c2)=O)CC2(CCC2)C1 c1(CNC(c2cccc(I)c2)=O)cccc(NC(C2CCOC2)=O)c1 S(=O)(=O)(c1cc(C)cnc1NCC1(CCO)CC1)NC(C(CC)C)C C(=O)(C1=CC2CCC(C1)C2)N1CCC(N(CC(COC)O)C)CC1 C1(NC(N2C(C(NOC)=O)CCC2)=O)CCN(C(=O)CN(C2CC2)CC)C1(C)C CC(C)CC(F)C(=O)NC1CCC(NC(=O)C(c2ccc(Cl)cc2)C)C1 c1(C(N(C(C)CCNC(=O)Cc2csnn2)C)=O)cnn2c1OCC2 CC(C)C(CCN(C)C(c1csc(Cl)c1Cl)=O)NC(=O)CCn1ccccc1=O c1(C(=O)NC2CC(CCNC(c3scc(C)c3)=O)C2)cc(C)nc(O)n1 C=C(C)CCC(=O)NC(C1CCCN1C(c1ccc(C2CC2)o1)=O)C c1(OC)ccc(S(=O)(=O)NCc2cc(C#N)n(C)c2)nc1 CCC(F)(F)C(=O)NC(C)CCNC(c1cn(-c2cnn(C)c2)cn1)=O N1(C(C(C(CC)C)C)=O)CCC(C2(O)CN(C(=O)CC3(C)CC3)C2)CC1 Cc1ccc(OCC(N2CC(CC(C)NC(C3CC(O)C3)=O)C2)=O)c(F)c1 CC1(C)CC(CC(N2CC(CO)C(O)C2)=O)CN1C(C1CC1C(F)F)=O C(=O)(C(CO)C(C)(C)C)NCc1c(C)ncc(Cl)c1 C1(C#CC(=O)NC2CCCC(NC(=O)C=C(C)C(C)(C)C)C2)(CC)CC1 Cc1ccc(C(=O)NCCCN(C)C(c2cnc(O)c(Cl)c2)=O)cc1Cl N1(C(c2c(C)n(CC(C)C)nc2)=O)CC(S)CC12CCOCC2 C1(c2ccc(Br)cc2)(NCC(n2cccn2)C)CCCC2(CCC2)C1 C1(C(=O)NC2CC2NC(C2CN3CCC2CC3)=O)C2(CCC2)C12CCC2 C1(CCNC(C(CC2CCC2)NC(C)=O)=O)CSCCN1C(c1cncs1)=O C1(NC(C(C)NC(c2cnc(S)nc2)=O)=O)CCCN(C)CC1 c1(SC)cc(C(N2CC(c3ocnc3CNC(c3nccs3)=O)C2)=O)ccn1 C(=O)(C(C)CC(C)(C)C)NC(C1N(C(C(C)NC(c2cccs2)=O)=O)CCC1)C c1(OC)ccc(C(=O)NC(C)CCCCNC(=O)CCc2cncs2)cc1 CCCCCCC(=O)N1CCC(NC(c2ccc(N)c(OC(F)(F)F)c2)=O)C1 CCCCC(CC)C(=O)N1CC=CC1CN(C(=O)C(C)(C)NC(=O)NCCC)C CC1(C)CC(CC(N2CCC3C(NC(c4c[nH]nc4Br)=O)C23)=O)CCO1 C1(NC(C2CC(=O)NC2)=O)CCCN(C(=O)CCc2nnc(C(F)F)o2)CC1 C=CCC(CC(C)C)C(=O)NC1(C2CN(C(c3cccnc3OC)=O)C2)CC1 c1(CC(=O)NC2CCN(C(CCSc3n(C)nnn3)=O)C2)ccccc1COC N12CCC(C)(C1)C2=O.C1(NC(=O)OC(C)(C)C)CCCC1NC(=O)C=C(Cl)Cl c1(OCC)nc(Cl)ccc1C(=O)NC1CN(C(=O)CCc2cccc(C#N)c2)C1 Cc1cc(-c2cn(CC3CC(CF)C3)nn2)cnc1C.C(=O)C(F)(F)C(C)O CC1CCCN(C(c2cnc(CNC(=O)COC3CC3)nc2)=O)C1CCO N1(C(CS(=O)(=O)N(C)C)=O)CC(C2CN(C(C3CCC(C(N)=O)C3)=O)C2)C1 N1(C(CC2N(C(c3c(N)nccn3)=O)CC2)=O)CCCCCCCC1 C1(NC(c2cc(CO)[nH]n2)=O)CCN(C(C2CC2C2CC2)=O)C12CC2 C1(C(=O)NC2CCCN(C(=O)Cc3c(F)cccc3F)C2)CCC2C(C1)C2(F)F c1(OCC)ccc(Cl)cc1CNC(=O)N(C(C)C(C)C)C1CC1 C(=O)(CC1OCc2ccccc21)N1C2CC(CC(NC(c3ccc(Cl)s3)=O)C2)C1 C1(C(=O)NC2C(NC(C(CCC)C(C)C)=O)CC2)C2CC3CC(C2)CC1C3 C(=O)(CCC(CC)NC(C1CC2CCC2C1)=O)NCCSCCC=C C(C)(CCC(=O)NCC1(F)CCN(C(=O)C=CCn2cncn2)C1)OC N1(C(C2C(CCC)C2)=O)CCC(CC(C)NC(C2CC(N(C)C)C2)=O)CC1 c1(CCC(=O)OC)ccc(C(=O)NCC(C)CNC(C2(C)CCOCC2)=O)cc1 N1(C(C(C)(C)OCC)=O)CCCC(CNC(c2cc(CF)on2)=O)CC1 C=CCCC(C)(C)C(=O)N1CC2(CCNC(=O)CC3CCN(C)C3)CCC1CC2 N1(C(CN2C(=O)C(C)C(C)C2=O)=O)CCC2CCN(C(C3(CF)CC3)=O)CC12 C1(NC(C2CC(C)(C)C2)=O)CCC(O)CN(C(=O)CCn2cncn2)C1 C1(CNC(COCC=C)=O)(CO)CCN(C(C2(C)CCOC2)=O)C1 N1(C(C2C(C)(C)C2)=O)CC(CO)C2(C1)CN(C(c1cc(F)ccc1O)=O)C2 CC(C)(C)C(CCO)NC(c1ccc(I)c(Cl)c1)=O O=C(CC1=CCCCC1)NC1(C(=O)NCC2(C3CCC3)CC2)CC(F)C1 N#Cc1cccc(NC(=O)COC(c2scnc2C2CC2)=O)c1 S(=O)(=O)(c1ccc(NCC2(CC#N)CC2)c(Cl)c1)N1C(CF)CC(OC)C1 C1(NC(c2c(CC)scn2)=O)CC2CC(NC(c3cc(Cl)no3)=O)C2C1 C1(OC)CCC2(C(=O)NCC3(NC(=O)CCC4CCCCCC4)CCC3)CC12 c1(CC)ncc(C(N2CC3C(C(=O)NCc4cnsc4)C3C2)=O)cn1 C(CCOC)(C(=O)N1CC(OC)C(O)C1)NC(c1cc(OC)n[nH]1)=O C(=O)(C1=CC(C)(C)C1)N1CC(SC)C(NC(C2(CN(C)C)CC2)=O)C1 Nc1ccc(C(=O)NCCNC(=O)CC2CCC(C(F)(F)F)O2)c2cnccc12 c1(C(c2nnnn2C)N)csc(C2CC2)n1.c1csc(CCCOc2ccccc2)c1 Cc1cc(C(=O)NCCCN(C(=O)C(C)(C)c2cccnc2)C)c(C)cc1Cl N1(C(CCC2C(C)=NOC2=O)=O)CC(N(C)C(c2c[nH]ccc2=O)=O)C(C)(C)C1 Cc1sc2ncc(C(=O)NC(C)CN(C)C(C3CC34CCOC4)=O)n2c1C CN1CCN(C(C2C=CC(NC(C3CCC(C)(C)CC3)=O)C2)=O)CC(O)C1 CC1CN(C(c2ccno2)=O)CCC1NC(=O)CC1CCC(=O)C1 c1cc2c(N3CCCC4(CC4)C3)[nH]c(=NCCC3(CC4CC4)CCC3)nc2s1 c1(OCC(=O)NCCCC(C)NC(C2(C#C)CC2)=O)ccc(C(F)(F)F)cn1 CC(CC(C)(C)C)C(=O)NCCN1CCC(NC(=O)COC2CC2)CC1 c1(C(N2CCC(C)(NC(c3c(CC)scc3)=O)C2)=O)ccccc1N=S(C)(C)=O c1(C(=O)NCCCN2CCN(C(C(COC)O)=O)CC2)cccc2oc(=N)[nH]c12 N1(C(C(C(=O)OC)OC)=O)CCC2(CC1)CC2C(=O)NCCN=S(C)(C)=O c1(C(=O)NCc2occ(C(=O)NCC(COC)O)c2)nccc(C)c1F C(=O)(CC1COCc2ccccc21)NC12CN(C(CNC(C)=O)=O)C(CC1)CC2 CC1(F)CCC(C(=O)NC2CN(C(C3CN(CC(F)(F)F)C3)=O)C2)CC1 C(=O)(C(C(C)(C)C)OC)NC1CCCN(C(c2n(CC=C)ccc2)=O)C1 CC(C)(C)C(C(=O)N1CCC1CNC(C1CC1C(F)(F)F)=O)c1cc[nH]n1 C1(NC(C(C)(C)OCC)=O)CN(C(c2cnn(C)c2SC)=O)CCC1C C1(O)(C(=O)NCC#CCNC(c2ccc(Cl)cn2)=O)Cc2ccccc2C1 C1(NC(c2csc(F)c2)=O)CN(C(C2CCC2(F)F)=O)C2CCCC12 C1(NC(C(CC(N)=O)O)=O)CC2CCC(C1)N2C(c1cccc(Br)c1O)=O c1(CC(=O)NCCC2(O)CCN(C(=O)CC3(C(F)F)CC3)C2)cncc(O)c1 N1(C(C(COC)C)=O)CCC(C(=O)N(CC(C)C(F)(F)F)C)CC1 N1(C(c2n(COC)ncc2)=O)CC2CCC(C1)C2NC(=O)CS(=O)C(F)(F)F CCCCC(O)C(C)C(=O)N1CC(OC)C(NC(c2cc(C3(C)CC3)n[nH]2)=O)C1 CCC(CC)(CO)C(=O)NCCN1CCN(C2CCN(C(=O)C(C)(C)F)CC2)CC1 C1(CC)CN(C(=O)Cn2nccn2)CCN1C(=O)C(CC=C(C)C)c1ccccc1 C1(CC(N2C(CN(C(C(C)OCC#C)=O)CC)CCC2)=O)(OC)CCOCC1 O=C(CCCc1cncs1)OCCSC1CCOC1 C#CCCCCC(=O)N(C(C)CN(C)C(c1cn(C2CCOC2)nc1C)=O)C c1(C(N(C2CCCN(C(CC3(C=C)CC3)=O)C2)C)=O)nnc2n1CC(=C)S2 c1(C(=O)NCCN(C(=O)C(=O)NCC2CC2)CC)csc(Br)c1 N1(C(C(C)OCCOC)=O)CC(C(=O)NCc2conc2C)OC(C)C1 c1(CNC(C2C(OC(C)=O)C2)=O)cccnc1C(F)(F)F N1(CCCC)CCC(CCOC)(N(C(=O)Cc2cc(=O)n(CC(C)C)[nH]2)CC)CC1 C(=O)(C(C)(C)CC(C)(C)C)NCC1CN(C(Cc2ccn(C)n2)=O)CC(C)(C)C1 N1(C(C2(SC)CC2)=O)CC(NC(=O)C(c2ccccc2)OC(C)C)C(C)(C)C1 C1(C(=O)NCCC(C)NC(=O)C2=CCCSC2)CC12CC(F)(F)C2 C1(C(=O)NCC2CCN2C(C2CC(=O)N(C(F)(F)F)C2)=O)CC2(CCCCO2)C1 CC(C)CC(CN=c1[nH]c2cc(F)ccc2o1)NC(c1ccc(F)o1)=O c1(C(C)O)nccc(C2(Cl)CC2)n1.C12(CCCC1)CC(=O)N2.C1(NC=O)(C)CC1 Cc1cc(=O)c(C(=O)NCCN(C(=O)CN(C)CCO)C2CC2)cn1C CCCCCCn1nnnc1C1(NC(C)C(C)SC)CC(n2ccnn2)C1 C1(CN(C)C(c2nccnc2C(N)=O)=O)CCN(C(C2C3COCC23)=O)CC1 N1(C(CCC=C=C)=O)CC(NC(=O)COC2CCC(F)(F)CC2)CC12CCC2 C1(O)(CN(C(=O)C(=O)NCC(F)(F)F)C)CN(C(=O)C(C)(C)c2cncnc2)C1 N1(C(C(CCC(C)C)NC(Cc2c(C)cccc2)=O)=O)CCc2ccccc2C1 CC1(C)CCCN(C(c2ccc(=N)[nH]n2)=O)C1C(N1CCSCC1CO)=O CN1CCN(C(C2(C#N)CC23CCC3)=O)CC1CNC(=O)C1=CCCC1 C(c1c(Cl)nc2ccccn12)=CC(=O)NC1CN(C(CC2CC(C)C2)=O)CC1O c1(C(N2C3(C(=O)NCc4n(C)cnc4)CC3CC2)=O)cn2c(n1)CCC2 C(=O)(C(C)C(O)CC(C)C)N1CCC(=C)CC1C(N1CC2(CCC2(C)C)C1)=O N1(CC(=O)N(c2nccs2)CC)CCC(NC(C2CC2CC)=O)CC1 CC(N=c1[nH]c(=NCC2CCS(=O)(=O)C2)[nH]c2ccsc12)c1ncc[nH]1 C1(C)(C(=O)NCc2cc(C3CCN(C(CC=C)=O)CC3)no2)CCCCNC1=O Cc1ncc(CNC(c2ccccn2)CN2CCCCC2)c(O)n1 CC1(CNC(c2c[nH]cc(Cl)c2=O)=O)Cc2ccccc21 C(=O)(C(C)(C)CCS(C)(=O)=O)NCC(CO)NC(CSC)=O c1(OCC(=O)NCCCN(C(CCCC)=O)CC)ccnc(C(F)(F)F)c1 C(c1ccc(Cl)cc1Cl)=CC(=O)NC1(CCO)CN(C(CN(C(C)=O)C)=O)C1 n1(CC)cc(C(=O)NCCCCNC(=O)CCCC2CCCC2)c(C(C)C)n1 c1(COC)ccccc1C(=O)NC(C)(CNC(c1sccc1CO)=O)C1CCC1 c1(C(c2nnnn2CCOCC)NCC=CC)c(C)noc1CC c1(C(=O)NCCCCNC(Cn2nnc(C)n2)=O)ccc(O)nc1Cl c1(C(N2CC(OCCC(N3C(C)(CCCO)CCC3)=O)C2)=O)cc(F)ccc1O c1(OC(c2cccc(CCN(C)C)c2)=O)cncc(F)c1Br C1(NC(C(C)(C)NC(C(CCC)C#N)=O)=O)CCOC2(CCC2)C1 c1(C(=O)NCCC(C)NC(C(N2C(C)CCCC2C)=O)=O)ccc(Cl)c(C#N)n1 c1(C(=O)NCC(C)(O)CNC(C2CC2F)=O)cnc(O)n(C2CC2)c1=O C=CCCC(C)(C)C(=O)NC1CC(C(F)C(=O)NCCCCC(C)(C)C)C1 C#CCC(C(N)=O)NC(C1(CC#C)CCN(C(c2cc(OC)n[nH]2)=O)C1)=O c1(SCC)ccccc1CC(=O)NC1CCCC1NC(=O)CC1CCCCO1 N1(C(COC(c2scc(OCC)c2)=O)=O)CC23CCCC2(C1)CN(C(=O)NC)C3 C1(C(N(C)Cc2cncnc2)=O)CCCCC1C1CC1 c1(C(=O)NCC(CNC(C2(NC(N)=O)CC2)=O)O)cc(C(N)=O)ccc1Cl Cc1ccc2cccc(CNCc3c(Cl)cccc3Cl)c2c1 C1(CC)CN(C(=O)Nc2ccccn2)CCN1C(c1ccc(=O)oc1)=O N1(C(CCCOC)=O)C2CCC1CC(C(=O)NC(c1ccc(C)cn1)C)C2 Cc1cc(CN2CCCCC2C(=O)Nc2ncc(Br)nc2CO)c(C)cc1Br CC1CN(N2CC3CCN(C(=O)OC(C)(C)C)C3C2)CC1C(F)(F)F CC1OCCC1(C)C(N1CC(O)(CCNC(c2cnn(C)c2Br)=O)C1)=O C(=O)(C(CC)C(F)(F)F)NC(CCCCNC(CCc1cccc(C#C)c1)=O)C c1(NCCN(C(=O)CCC2CC(C)(C)CO2)OCC)cccc(OC)c1[N+](=O)[O-] N1(C(c2nc(C)sc2)=O)CCC2C(CCCN2C(=O)COCC2CCC2)C1 C(C(C)(C)C(=O)N(CC(C)CNC(=O)Cn1cccn1)C)OC(C)C C1(NC(c2ccc(OCCC#C)cc2)=O)C2CC1N(C(c1cnn[nH]1)=O)C2C N1(C(C(C(CC)C)O)=O)CCN(C(=O)C(C)N(C)C)C2COCC12 C1(C(=O)NC(CNC(c2n(C(C)C)ccn2)=O)C(C)C)Cc2cccc(F)c2O1 c1(OC)c(C)cc(C(=O)NC2CCN(S(=O)(=O)c3cccnc3)CC2F)cc1C N1(C(COCC(C)C)=O)CCOC(C(=O)NC(c2ncc[nH]2)CO)C1 CC1CN(C(C2(Oc3ccccc3)CC2)=O)CC1CNC(C1(CCCl)CC1)=O Cc1cc(CNC(C2CCCCN(C(=O)C3=C(Cl)CCC3)C2)=O)cc(F)c1 C1(NC(C2C(C)C2)=O)CCN(CCNC(=O)CC(C)c2cnn(C)c2)CC1 Cc1cc(F)c(C(=O)OC(C)(C)C)cc1Cl.N12CC(C1)CS(=O)(=O)NC2=O c1(C(=O)NC(C)C(C)NC(c2cscc2C(N)=O)=O)nnn2c1C(=O)NCC2 N1(C(C(F)=CCC)=O)CC2CCOC2(CNC(=O)C(C)CC(N)=O)C1 N1(Cc2ccc(C#C)s2)CCN(C(=O)CCCCC)C2CC12 CC1COCCC1CNC(c1ccc(CNC(C2C3CC4C(C3)C24)=O)s1)=O N1(C(C23CC(C)C2C3)=O)CC(CNC(=O)C(C)(C)n2cnnn2)CC(C)(C)C1 N1(C(C(C)=C2CCC2)=O)CCN(C(=O)CC2CCCOC2)C(CO)C1 c1(C(C)=O)cccc(-c2cn(CC3CN(C(=O)CCC4CCCCO4)C3)nn2)c1 C=CC(O)C(=O)N(CCNC(=O)Cc1cnc(C)s1)CCc1ccccc1 c1(C(CNC(C2C(OC)CC2)=O)NC(=O)C=Cc2ccco2)ccccc1F C1(C(=O)NC2CC3CC(NC(c4cccnc4)=O)CC32)CN=C2N=CNN2C1 S(=O)(=O)(c1csc(C(=O)NC2CC(O)CN(C(=O)Cn3ncnn3)C2)c1)NC C1(C(=O)NCC(N2CCN(C(C3(C)CC3(F)F)=O)CC2)C)CC2C=CC1C2 N1(C(c2c(COC)ncs2)=O)CCC(C)N(C(C23CCC(OC)(CC2)C3)=O)CC1 n1(CC)ccc(CCNC(c2ccsc2C)c2nnnn2CC2CCOC2)n1 C(=O)(CCC1(NC(=O)C(F)C2CCCC2)CCC1)NC(c1cc[nH]n1)C c1(CC)nc(C)c(C(=O)NC2CC(CNC(c3cnn(CCO)c3)=O)C2(C)C)o1 Cc1nnc2ccc(CCn3cc(CN(CCC#N)CCO)nn3)nn12 Cc1cc(CNC(c2ccnc(O)c2)=O)oc1C(=O)NCc1cnn(C)c1O N1(Cc2cc(C)[nH]c2C)CC2CCC1CN(C(=O)C(=O)c1ccco1)C2 CCC(C)CC(C)C(=O)N1CCC(NC(c2ccc(CO)nc2)=O)C(C)(C)C1 C(=O)(N=c1nc(C2CCCCN2C(=O)Cn2cncn2)[nH][nH]1)C(=O)OC(C)(C)C CCC(CNC(c1cc(CNC(c2cc(C)c[nH]2)=O)ccn1)=O)C(C)C c1(CC)cc(C(=O)NCC2(C)CCC(NC(=O)CNC(=O)C(C)(C)C)C2)ccn1 C(=O)(C(CC(C)CC)NC(C1CC2(CCC2)CO1)=O)NCc1cnc(CC)[nH]1 c1(C(N2CCC(C)(CNC(c3cc(CO)[nH]n3)=O)C2)=O)ccc(F)cc1F c1(OC)coc(C(=O)NCC2CC(C)(C)CN2C(=O)CN2CC3CC3C2)cc1=O c1(C(=O)NC(C2CN(C(C3C4COCC34)=O)C2)C)noc2cc(Cl)ccc12 C1(CNC(C2C(NC(c3ncc(OC)nc3)=O)CCO2)=O)CCOC(C)(C)C1 c1(CN2CC(CC(=O)OC)OC(C)C2)cc2cc(Cl)cnc2o1 C1(C(N2CC(CN(C(c3cc(OC)n(C)n3)=O)C)C2)=O)CC12CCOCC2 N1(C(c2c(C)onc2O)=O)C2CCCC1CC(NC(c1cn(CCF)nn1)=O)C2 C=CCCN=C(NCc1ccc(C)nc1OC)NCC1CC(CC)C1 C12(NC(C=CC=CC)=O)CCC(CNC(c3cc(C)c(OC)c(C)c3)=O)(CC1)OC2 CCC(Cc1ccccc1)C(=O)NC1CN(C(C23CC(CN2C2CC2)C3)=O)CC1O CC1(C)CC=C(C(=O)N2CCC(C)(CNC(=O)CC(CN(C)C)C(F)F)C2)CC1 c1(OC)ccc(Br)c(S(=O)(=O)N2CCc3nc(-c4ccccc4)ncc3C2)c1 N1(C(Cn2c(C)nnn2)=O)CC2C(NC(=O)C3=COCC3)C2C1 c1(C(C)NC(C2(CC(C)=O)CC2)=O)nocc1C(=O)NC(c1ncc[nH]1)C C(C(C)CCCC(C)C)NC(C1(NC(c2c(COC)cc[nH]2)=O)CC(O)C1)=O C1(NC(C2CC2c2ccccc2)=O)CCN(CC2CCC2)C1 CC1CCCC1C(=O)CNC(=O)C(C)OC(C1CCCN1C(=O)OC1CCC1)=O C1(CNC(c2ccc(C(C)C)o2)=O)CCC2(CN(C(=O)C(O)c3ccco3)C2)O1 c1(N(C)CC2CCN(C(=O)C=Cc3cn[nH]c3)C2)cc(C(N)=O)nc(Cl)n1 CC(C)CC(CNC(C1CCS1(=O)=O)=O)NC(=O)CC1(C(F)F)CC1 N1(C(C=CC)=O)CCN(C(=O)C(N2CCC(O)CC2)C)CC(C)(C)C1 Cn1[nH]c(=NC(=O)C2CC2C2CN(C(c3cnnc(O)c3)=O)C2)cc1C(N)=O c1(NC(C(C)OC(c2cnc(SC)s2)=O)=O)cccc(N2CCOC2=O)c1 N1(C(C2N(C)CCC2)=O)CC(NC(c2cnc3[nH]nnc3c2)=O)C2CCCCC12 C1(OC)CCCCC1NC(C1(C(=O)NCC2(OC)CCCCC2)CC1)=O C1(C2CN(C(=O)C(n3cc(C)cn3)C)C2)(NC(c2cn(CCOC)nn2)=O)CC1 N1(C(C2(C)CC3(CCC3)C2)=O)CCC2(CCN(C(c3cc(C4CC4)ns3)=O)C2)C1 C(C(CNC(c1ccc(CSC(F)F)o1)=O)C(F)(F)F)NC(C1CC(C)(O)C1)=O N1(C(c2c(C)cc(C#N)cn2)=O)CC2(C=C(C(=O)NCC3CCC4CC34)CO2)C1 C12(C(=O)NC(C)C(C)(O)Cc3cccc(Br)c3)CC3CC(CC(C3)C1N)C2 CCC(CC)(CO)C(=O)NC1COC2(CNC(=O)CC(C)C)CC1C2 C1(CNC(C(C)OCCOC)=O)CCC(C(=O)NCCC(O)C2CC2)C1 c1(C(CNC(=O)CC2CCC(O)C2)NC(CC2(N(C)C)COC2)=O)ccc(F)cc1 N1(C(C(CCC)C#N)=O)Cc2n[nH]cc2C1C(=O)NCc1cccc(F)c1F c1(C(=O)NC23C(CCN(C(CCC#CC)=O)CC2)C3)ccc2nn(C)cc2c1 C(=O)(CC1=CCCCC1)NCC1C2N(C(C=C(CCN(C)C)Cl)=O)C(CC2)C1 C1(NC(c2cc(C(N)=O)sc2)=O)COC2(C1)CN(CC1CCCOC1)C2 C12(C(=O)NCCCCNC(c3csc(Cl)n3)=O)CCCC1CC2 C(=O)(CCC(C)(C)NC(C1CCCOC1C)=O)N(CC#C)CCF C#CCC(O)C(=O)NC1CC(N(C(=O)C(c2ncc(Cl)n2C)(F)F)C)C1 C#Cc1cccc(CC(=O)NCCCC(=O)Nc2ccccc2C#C)c1 O=C(C1COc2ccccc21)NCC1CC(O)CN1C(c1cc(O)ncn1)=O c1(OCC)cccc(C(=O)NC(C)(C)CCCNC(=O)CCC2CCOC2)c1N C(=O)(CCCC(C)(C)CC)NC1CC2CN(C(C3(CCCC)CC3)=O)CC2C1 N1(C(C=C(C)I)=O)CC2C(NC(c3cc[nH]n3)=O)C2C1 CCC1=NOC(CC(N2CCCCCC2)=O)C1.N12CCC(C1)OCC2=O CC(O)CCCC(=O)N1CCCC1(C)CNC(C1CC2C=CC1C2)=O N1(C(C(C)=CC)=O)CC2CCN(C(c3csc(N4CCC(O)CC4)n3)=O)CC2C1 c1(C(NNC(N2CCCC(CC(C(=O)OC)N)C2)=O)=O)ccc(S(N)(=O)=O)s1 c1(NC(c2cnc(Cl)n2C)c2n(CC=C)nnn2)ccc2oc(CSC)nc2c1 c1(C(C)NC(C23CCCN(CCC2)C3)=O)cccc2ccccc12 N1(C(c2nnn(C)n2)=O)CCC2CCN(C(C3(O)CCC3)=O)CC12 CCCCCC(O)C(=O)NC(CNC(c1cn(-c2ccc(Cl)cc2)nn1)=O)CO N1(C(C(C)(C)OC)=O)CCCC(C)(CNC(c2ccc(O)c(CO)c2)=O)C1 C=C(C)C(CC(=O)N(CCCN(C(=O)CC1CC2CC2C1)C)C)OCC c1(C(N2CC(O)(CCNC(CCCCC(N)=O)=O)C2)=O)cc(Cl)cc2c1CCC2 C1(C2CCCN(C(C3(CF)CCC3)=O)C2)(NC(c2cc(C)c(=O)n(C)c2)=O)CC1 C12(CNC(Cc3nc(C)cc(OC)n3)=O)CCCC1N(C(=O)CNC(C)=O)CCC2 C1(NC(CC2(C)CCCC2)=O)CCCCC1CNC(=O)CN1CSCCSC1 c1(CN(C(C=CCC)=O)C)ccc(CNC(=O)C(CC)OC2CC2)cc1 C(CCS(=O)(=O)C(C)(C)C)NC(C(CCC)CC)c1nnnn1C(C)(C)CC c1(OC)ccccc1C(C)=CC(=O)NC(C)CCN(C)C(C1(F)CC1)=O C(=O)(C(C)CC(C)C)NC(c1cccc(OC)c1)CNC(C1(C)CCC(=O)C1)=O CC(C)C(O)C(C)C(=O)N1CC2(C(=O)NC(C(C)(C)O)C3CC3)CC1CO2 C1(NC(CCSC)=O)CCN(C(c2ccc3c(c2)C(C)CO3)=O)CC(C)(C)C1 C=CCCCC(C)(C)C(=O)NCC1CN(C(=O)CCc2nccn2C)C2CC12 N1(C(CNS(CCOC(C)(C)C)(=O)=O)=O)CC(=O)CC1C(=O)NC1CC1 Cc1ccc(C(=O)NCC2CN(C(c3ccsc3C(F)F)=O)CCO2)c(O)c1 c1(C(=O)NC(CNC(CC2C(C)CCC2)=O)(C)C)cnc2cnc(Cl)cc2c1 c1(OC)ccc(C)cc1C(=O)NCc1cccc(NC(C2CCC(F)C2)=O)c1 C1(CNC(C(c2ccccc2)N(C)C)=O)C=CCN1C(c1cnc(Cl)s1)=O C12(NC(COCC)=O)CCOCC1CN(C(=O)CCc1ccc(Br)cn1)C2 C(=O)(C(O)C(F)(F)F)NC(C1N(C(CC2(CC(=O)OC)CC2)=O)CCC1)C C1(CC)C2CCN(C(=O)C(C)=CCNC(=O)COC3CCOCC3)CC12 C(=O)(C1=CCCC(C)(C)C1)N(C)CC1N(C(C(C(C)C)CO)=O)CCOC1 CCCS(=O)(=O)CC(=O)N(C1CCCN(C(c2ccc3oncc3c2)=O)C1)C CC1(C)CCOC(C(N2CCN(C(=O)COCc3nc[nH]n3)CC2CO)=O)C1 C(CCc1ccccc1)(CN=C(NC1CCC1)N1CC2CC1CS2(=O)=O)SC C=CCC(C(=O)N1CCN(c2nc3ccccc3o2)C(C)C1)C(C)C N1(C(CC(C)C)=O)CC2(CCC2CNC(=O)Cc2cn[nH]c2)C1 N1(C(C(C)=C(C)C)=O)CCCC1C1(NC(C2CC(C)(O)C2)=O)CC1 c1(C(=O)NC(CC)(C)c2nn[nH]n2)cnn(Cc2ccccc2)c1Cl C1(C(=O)NC2CC3(C(NC(Cc4ccc(OC)cc4)=O)C3)C2)CC2(C1)CC(O)C2 c1(OCCCC(=O)NC(CC)CN(C)C(C2(F)CC2)=O)ccc(Cl)cc1C N1(C(c2c(CC)[nH]cc2)=O)CC(NC(=O)CCC2CC2(Cl)Cl)CC2(CC2)C1 CCC(C)(COC)C(=O)N1CCCC(C(C)C(=O)NCCCOC(C)=O)C1 S(=O)(=O)(c1cn[nH]c1)N1CCCC(C(=O)OC(COC)CN2CCOCC2)C1 c1(C(=O)NCC(CNC(=O)C(C2(O)CCCC2)F)OC)snnc1C1CC1 n1(C2CN(C(CCCn3cc(C=CC)nn3)=O)C2)cnc2ccccc2c1=O C1(CNC(C)=O)CN(C(=O)C=Cc2ccnn2C(C)C)CC2(CCC2)O1 c1(CNC(c2cccc(N3CCNCC3)n2)=O)cc(Cl)c(Br)cc1Cl C1(NC(Cc2cc(C)on2)=O)CN(C(c2cnc3scc(C)n23)=O)CC12CCC2 c1(NCC)cccc(C(=O)NC2CCC(NC(C3CCN(C)C3=O)=O)CC2)c1 N1(C(COCCC)=O)CCC2(CCCC2NC(C2CC3C=CC2C3)=O)CC1 C1(C)(CNC(c2c(COC)ccs2)=O)CN(C(c2ccccc2C)=O)CCO1 C1(CC(=O)NC2(CN(C(C(C(C)C)SCC)=O)C)CC2)CSc2ccccc2O1 c1(C(=O)NCC2(NC(C=NOC)=O)CC2)cc(NC)ccc1Cl C1(COC)CN(C(C2CCC(NC(C3C(C)(C)C3(C)C)=O)C2)=O)CCO1 CC1CC(N=c2nc3c(cnn3C)c(NCCc3ccn(C)n3)[nH]2)CCS1 c1(C(N(CCNC(c2occc2C)=O)CC)=O)cc2ccc(OCC)cc2cn1 N1(C(C(OCC)OCC)=O)CCCC1C(=O)N(C(C)C)CC1CCCOC1 C#CCCCC(C)C(=O)N1CCC(C(N2CC(C(C)(C)O)C2)=O)C12CC2 c1(C(N(C2CCC(NC(C=CC)=O)CC2)C)=O)nc(OC)ccc1F C(C(F)(F)C(F)F)NC(C(CC1CC1)OC)=O.C1(=O)C=CC(=O)NCCN1 C(=O)(C(CC(C)C)NC(C1CC(C(C)C)=NO1)=O)N(CC#C)CC c1(CNC(=O)C2CC2)ccncc1OC1CCN(C(c2cc(C3CC3)[nH]n2)=O)C1 c1(C(=O)NCC(CCOC)NC(C2(NCC)CCC2)=O)cc(C(F)F)ccn1 N1(C(c2oc(CC)c(C)c2)=O)CC2CC(C)N(C(=O)C(COC)CC(C)C)C2C1 Oc1c(-c2nc(-c3cc[nH]n3)nn2C2CCOCC2)ccc2c1CCCC2 CC1=CCC(C)(C(=O)NCC2(C)CC(NC(=O)CC(=O)OC(C)(C)C)C2)CC1 c1(C(N2CC(CNC(CC(CC)C)=O)C(C(F)(F)F)C2)=O)ccc(F)c(Cl)n1 Cn1nnnc1N1CCC(NC(C2CN(S(=O)(=O)C(F)F)C2)=O)C1 N1(CC(=O)N(CCOCCCNC(C2C(=C)C2)=O)C)CCNC(=O)C1 c1(C(N(C(CC)CNC(=O)CSS(C)(=O)=O)C)=O)ccc2nc[nH]c2n1 c1(OCCC(=O)NCCNC(c2ccccc2Br)=O)ccc(F)c(Cl)c1 N1(C(c2ccc(SC)cc2)=O)CCC(C)C(CNC(C2CC=C(C)CC2)=O)C1 CCC(C)CC(C)C(=O)NC1CC(NC(c2ccccc2NCCO)=O)C1 CS(=O)(=O)c1ccc(NC(=O)C(=O)NC23CC4CC2C3C4)cc1C(F)F C1(CNC(CSCC=C)=O)C(CNC(=O)CC2OCCCO2)C1(F)F c1(C(C)C)nnnn1CC(=O)NC(C)CCN(C(=O)Cn1ccc(C2CC2)n1)CC O=C(C(O)CC1CC1)NCC1(F)CC(NC(C23COCC2C3)=O)C1 c1(C(=O)NC2C(OC)CN(C(=O)CCC(C)C)C2)cc2ccc(F)c(F)c2o1 C1(C(=O)NC(C2CCN(C(c3ccc(CN(C)C)o3)=O)C2)C)CCOC1C(F)F c1(NC(C(C)C)CCN(C)C(c2cc3n(n2)CCC3)=O)cc(S(C)(=O)=O)ncn1 N1(C(CN(C(=O)Cc2cnoc2)CC#C)=O)CC2CCOC2C1 c1(SCC(N2CCC(CNC(CSC(C)C)=O)C2(C)C)=O)ccc2c(c1)CCC2 c1(CC(=O)NCC(C)(C2CCC2)NC(C2CC2F)=O)ccc2cccnc2c1 c1(NC)cccc(C(=O)N(CC(C)NC(c2ccnc(C(C)(C)C)c2)=O)C)n1 c1(C(=O)NCCC2(O)CN(C(c3nc(OCC)sn3)=O)C2)cnc(C)nc1C C1(CNC(CC=C=C)=O)CCC(C)N(C(c2ccc(NCCO)cc2)=O)C1 CCC(C)C(O)C(=O)NCC1CC(F)(F)CN1C(c1cc2occc2[nH]1)=O c1(C(=O)NC2(CO)CCCN(C(CSCCN(C)C)=O)C2)ccc2occc2n1 C1(NS(C)(=O)=O)CCC(C(=O)NCCn2ccnn2)C1.N1(CCO)CCOCC1 C1(OC)CCCCC1C(=O)NCCCCCN(C)C(C1(N=[N+]=[N-])CC1)=O CC(C)(C(=O)NCc1cn(C2CN(C(C3(F)CCOC3)=O)C2)nn1)C(F)F C1(C(N(C)CCNC(C2CC(F)C2)=O)=O)SCCN1C(=O)OC(C)(C)C Cc1ncnc(C(=O)NCCC2(C(=O)NCCC(C)(C)C)CCC2)c1C c1(C(N2C(C(=O)NCC)CCC2)=O)ccc(C(N2CC(C(C)SCCC)C2)=O)o1 C(=O)(CC(C)(C)C(F)F)N1CCC(NC(CC(C)c2ccco2)=O)(CO)C1 N1(C(C=COCC)=O)CC2CCC2(CNC(C2CC23CCCCC3)=O)C1 C1(CNC(C(CCO)N(C)C)=O)CN(C(C2(C(C)(F)F)CCC2)=O)CCC1(C)C n1(CCC(=O)NCCNC(C2(CCC)CC2)=O)nc(O)c2ccccc12 C1(NC(c2cccc(C(C)C)n2)=O)CC2CCC1N2C(=O)COCC1CC1 C(=O)(C1=CCN(C(C2CC2CC(C)C)=O)CC1)N(CC(CC)OC)C C1(CNC(C2CC(O)CN2C(=O)CCC2CCCO2)=O)CC2(CCCO2)C1 c1(C(=O)NCC(CNC2CC(C(=O)OC)C2)(C)C)oc2c(OC)cccc2c1C c1(CNC(C(c2ccccn2)C)=O)ncc(C(F)F)cn1 Cc1nc(C)n(CC(=O)NCc2nc(C(=O)NC3CCOC3=O)co2)n1 N1(C(C(CCC)OC)=O)CC(C2CC2)(C(=O)NCCCCCCC2CC2)C1 C1(c2cn(C3CC(OCC)CC3O)nn2)C=CCC(C(=O)NC(=O)C2CC2)C1 C1(C(=O)NC(c2cn(C)nn2)C)CCN(C(=O)CC2CCOCC2)C1C C1(C)(NC(Cc2cnc(C)s2)=O)CCC(NC(=O)CCC(C)(C)N(C)C)CC1 C1(NC(c2n(CCC)ncc2)=O)CCN(C(c2csnc2C)=O)CC1CO N1(C(CCC(=C)Cl)=O)CC(NC(=O)CCCc2ccncc2)CC12CCOCC2 Cc1[nH]nc(C(F)(F)F)c1C(=O)NC1C2CC1N(C(C1CCS(=O)(=O)C1)=O)C2 C1(C(N2CCCC(CNC(c3ccn(C)c(=O)c3)=O)C2)=O)CCOCC12CCC2 N1(C(c2c(OC)cccc2)=O)CCCC(O)(CNC(c2ccoc2C(C)C)=O)C1 c1(C(N2CC3C(CNC(C45CC(CO4)C5)=O)C3C2)=O)ccc2cnsc2c1 c1(OC)ccc(F)c(NC(C2(NS(C)(=O)=O)CC2)=O)c1F.N12CCN(CC1)CC2 C(=O)(CCCC(N)=O)NCCC(C)NC(CCC(C)OCC)=O c1(OCC)cc(C(N2CC(C)(NC(C3CCCSC3)=O)C2)=O)cc(F)c1 c1(C(=O)NC(C)CCCNC(=O)CC2CCCOCC2)cnc2n1CCC2 C1(NC(c2cncc(N=[N+]=[N-])c2)=O)CCCCC12CCN(C(C1CCCS1)=O)C2 CC1CN(C(C2C=CCC2)=O)CCCN1C(c1ccnn(C)c1=O)=O C1(NC(c2cc(C)c(Cl)s2)=O)C2CC3CN(C(=O)CC4CCCC(O)C4)C1C3C2 Cc1cc(C(=O)OC(C2CCCN(C(=O)OC(C)(C)C)C2)C)c(Cl)cc1F c1(-c2cncc(CNCc3n(C)c(=O)ccc3)n2)cccc(C#N)c1F C1(CNC(=O)NCC(C)N(C(=O)OC(C)(C)C)CC)CCCN(C)C1 c12nc(CC3CC3)nn1-c1ccc(cc1)C2.N1(CCOC(C)=O)CCCC1 C1(NC(c2cccc(CNC(c3ccn(CCF)n3)=O)n2)=O)CC2(CCCO2)C1 C=CCC(CC(C)C)C(=O)N1CCCC(CNC(c2cc(C)c(C)c(F)c2)=O)C1 c1(CC)ccc(F)cc1C(=O)NCCNC(=O)C=Cc1ccc(C(N)=O)o1 c1(CN2CC(C(CC)=O)C(C)C2)ccc(Cl)c(NC(c2cncc(Br)c2)=O)c1 c1(SC)cc(C(=O)NCC23CC(NC(=O)CC=C(C)C)(C2)C3)c(Cl)cc1Cl N1(C(C2COCCN2CC(F)F)C)CC2(CNC(=O)N2)C1 C(C(C)(C)CNC(c1ncsc1C)=O)C1CN(C(C(C)NC(C)=O)=O)C1 N1(C(C)Cc2nc(Br)cs2)CCC2(CCN(Cc3ccccc3OCOC)C2)C1 O=C(C1=CCCCO1)NC1CCCC1N1CCN(C(C2CSCCS2)=O)CC1 C(=O)(C1=NOC2(CCC2)C1)N1C(C)CCC(NC(c2c(OC)cccn2)=O)C1 C1(NC(C2C=CCC2)=O)CC2CCC(C1)N2C(C1COC2COCC2O1)=O Cc1ccc(C(=O)NCC(N2CC(NC(=O)C(F)C(C)C)C2)=O)cc1 N1(C(C(CC(=O)OCC)C)=O)CC2(CCC(CNC(c3ncc[nH]3)=O)O2)C1 C1(C(N(CC(COC)O)C)=O)OCCC1NC(=O)CCCNC(=O)OC N1(C(C(C)SC(C)C)=O)CC(C2CC2)(C(=O)NCC2(C)CCC2)C1 c1(C(=O)NC2CC(CO)N(C(=O)CCC3CC(F)(F)C3)C2)c(Cl)cncc1Cl n1(CC(=O)NCCC2(NC(=O)CN3CCOCC3)CC2)nnc(-c2ccsc2)n1 C1(NC(CC(CCC)O)=O)CN(C(=O)C=C(C)C(C)C)C2(CCC2)C1 C1(OC)CCN(C(C2(OC)CCN(C(C3CCC4CC34)=O)C2)=O)C1C CC1CCCC1(C(=O)NCCC1CC=CC1)NC(c1nc(Cl)cs1)=O C(=O)(C(F)C(C)(C)O)N1C(C)(CC(=O)NCC2CCN(C)CC2)CC1 C1(NC(c2c(C)sc(Cl)n2)=O)CC2CC1N(C(=O)CCCc1cccnc1)C2 c1(-c2cn(C(C)C(=O)NC(c3ccns3)C)nn2)cccc(C(=O)O)c1 N1(C(c2c(C)nncc2)=O)CC(CNC(c2cc(O)ccc2F)=O)C(C)(C)C1 Cc1nc(-c2nc(-c3ccc(Cl)s3)nn2CC(C)(C)CO)c2n1CCCC2 C(=O)(C(O)C(C)CC)N(CCNC(=O)CCc1nc(SCC(F)(F)F)no1)CC c1(C(=O)NC2CC(N(C)C(c3cnn(C)c(=O)c3)=O)C2)ccc2c(ccn2C)c1 N1(C(C(COC)(C)OC)=O)CCOC2(CCN(C(C3(F)CCCCCC3)=O)C2)C1 c1(C(N)=O)cc(C(=O)NC2CCC(NC(C3CCCC3c3nc[nH]n3)=O)C2)on1 c1(C(=O)NCCSCC(=O)NCCC(CC)(C)O)c(C)ccnc1C N1(C(C2CC=C(C)CC2)=O)CCCC(F)(CNC(=O)Cc2ccc(CO)cc2)C1 c1(OC)ccc(Cl)c(C(=O)N(CC(C)CNC(=O)CCc2cnc(C)o2)C)c1N C1(C(=O)NCC(C)N(C)C(C2CC2[N+](=O)[O-])=O)C2C3CCC(C3)C12 CCCCC(C)C(=O)NCC(O)CNC(C1CSC1)=O Cc1c(C(N2CC(NC(c3cnc[nH]3)=O)CC2(C)C)=O)oc2ccc(Cl)cc12 Cc1csc(C)c1C(N1CC(C(=O)NCC2C(C)C2(F)F)C(C)C1)=O C#Cc1ccc(C(=O)N(CCC)CCNC(c2ccoc2CC)=O)c(OC)c1 c1(C(N2CCCC2C2(NC(C3(CO)CCOCC3)=O)CC2)=O)nccc(Cl)c1F C=CCC(CNC(=O)C(C)CC1CCC1)C(=O)NCCNS(N)(=O)=O n1(CC=C)nc(-c2ccoc2C)nc1-c1ccccc1Cl C12(NC(CSCCOC)=O)CCCC1N(C(=O)C(C(C)(C)C)SC)CC2 C1(C(=O)NCc2c(OC)nsc2)CCN(C(=O)CCc2ncccn2)C12CCC2 C(C1=CCCSC1)(c1nnnn1C)NCC1CC(OC(C)(C)C)C1(C)C c1(C(=O)OCC)cc(CNC(=O)NCC(c2cnccc2C)(C)C)cc(Br)c1 Cc1[nH]nc2c1CC(N=c1nc3c(cnn3C)c(NCCC(O)C(C)C)[nH]1)CC2 Cc1ccc(C(N2CC=CC2CNC(C2(Cl)CC23CCC3)=O)=O)nc1 c1(C(=O)NCC2CN(C(=O)CC3CC3)C2)cc(O)cc(O)c1 C1(C)(C(=O)NC2CCN(C(c3c(C)cnnc3)=O)C2C)COc2ccccc2O1 C1(C(=O)NCc2ccc(F)cc2)CC12CCN(Cc1ccc(Br)nc1Br)C2 c1(OC)ccc(C)c2[nH]c(C(=O)NC3CC(N(C)C(C4CCOC4=O)=O)C3)cc12 N1(C(c2cccc(CC)c2)=O)CC(C)CCC1CNC(C1CC(OC(F)F)C1)=O CCCCC(CC)C(=O)N1CCC(C2CC2)C1Cn1cc(CCOCCO)nn1 C1(N(C(=O)C=CC2CCCO2)C)CCN(C(=O)CCc2nccn2C)CC12CC2 C(=O)(C(CC(C)(C)C)OCC)N1CC(C(C(=O)NC2CC(O)(CC#C)C2)OC)C1 CCCCCCC(F)C(=O)Nc1cccc(CNC(=O)C(O)CCCC)c1 c1(C(=O)NC(C2CN(C(=O)COC3CC=CC3)CCO2)C)cccc2nsnc12 Cc1nc(C2CC2)oc1C(N1CC=CC1n1cc(CNN(C(C)C)C2CC2)nn1)=O C(C)(C)(CCC(=O)NCCC1(OC)CN(C(=O)C(C)(C)CO)C1)OC c1(OCC(=O)NC2C3CCN(C(c4nc(C)sc4)=O)C32)ccc(S(N)(=O)=O)cc1 c1(NCC(CC)N(C)C)[nH]c(=NCc2[nH]cnc2C)nc2c1ncn2C(C)C C1(C(=O)NCCCN(CCC)C(c2cnn(CC)c2)=O)CC2(CSC2)C1 C(=O)(C1CCCc2sccc21)N(CCNC(c1ccc(C)s1)=O)CC N1(C(c2cccc(C(F)F)n2)=O)CC2(C1)CN(C(=O)C(N1CCOCC1)O)C2 C1(CC)CC(C(N2CCC(CNC(=O)CC3CCCS3(=O)=O)CC2)=O)CC(=O)N1 c1(NC(Cn2nnc(C(N(C(C)=O)CC3CCN(CC)C3)=O)c2C)=O)ccc(CO)cc1 C12(NC(c3n(CCN(C)C)ncc3)=O)CCCC1N(c1ncncc1Cl)CC2 c1(NC(N2CC(CO)OC3(CCC3)C2)=O)ccc2ccc(O)nc2n1 C(CCCCC(=O)NC1CCN(C(C2(CF)CC3(CCC3)C2)=O)CC1C)OC N1(C(C23N(C(C4(O)CCSC4)=O)CC(C)(C2)C3)=O)CC(C2CCCCC2)C1 N1(C(CC2(C)CCC2)=O)CCC(C)(C)C1CC(=O)NC1(C)CCCC1(F)F C1(NC(C2C(C(=O)Nc3c(C(=O)OC)n[nH]c3)C2)=O)CC(=O)NC(=O)C1 N1(C(C(CCCNC(=O)CC2CC(F)C2)O)=O)CCC12CCC(O)CC2 C=C(Cl)CCC(=O)NC1CC(C(C)NC(=O)C(c2ccc(OC)cc2)=O)C1 C1(NC(C(C)n2cccn2)=O)CC(=O)N(C2CN(C(=O)CC3CCCC3)C2)C1 c1(OC)cc(C(=O)NCCCNC(=O)C(O)CC2CC2)cc(OC)c1OC(F)F c1(CCNC(C(n2cc(C(O)C3CC3)nn2)C)=O)ccccc1C1CC1 N1(C(CNC(N)=O)=O)CC(NC2CCN(C3CC3)C2=O)C2(CCC2)C1 Cc1ccc(C)c2[nH]c(C(=O)NC34CCCCC3OCC4)cc12 N1(C(=O)NCC2(F)CC(CC3CCC3)C2)CCSCC1c1ccccc1 C1(OC)CN(C(c2c[nH]nc2C(C)C)=O)CC1NC(=O)C(N1CCNC1=O)C c1(CCNC(c2c(C)nn(C)c2C)c2n(CCSC)nnn2)c(F)cccc1Cl C(C1=Cc2cc(Cl)ccc2OC1)=CC(=O)N(C1CCNCC1)CC#C C1(NC(c2ncn(C(C)(C)C)n2)=O)CC2CC1N(C(c1ccco1)=O)C2 CON(C)CCCNC(C1(NC(=O)CCOC2CCCOC2)CCCC1)=O C1(CN(C(C(=O)NCC=C)C2CCSC2)C)CCCCO1 N1(C(=O)Cn2ccc(C(F)(F)F)n2)CCOC(CNC(C2(O)CC(CF)C2)=O)C1 N1(C(c2cccc(CC)c2)=O)CC(NC(=O)COC(C)=O)CC12CCCC2 C1(F)(n2cc(-c3n(C)cnc3)nn2)CCC(NC(c2cc(CN)c(Cl)s2)=O)C1 C1(NC(C2C3CCN(C(CC4(OCC)CCC4)=O)CC32)=O)CCC(=O)N(C)C1=O C1(C(=O)NCC(CC)NC(=O)CCc2cccc(Cl)c2)CC2COCC2C1 C1(c2cccc(C3(C(N4CCC(C)CC4)=O)CCCC3)c2)OC(C)(C)C(C)(C)O1 c1(C(=O)NCC2(NC(C(C(C)OC)O)=O)CCC2)ccccc1[N+](=O)[O-] N1(C(c2c(C(N)=O)coc2)=O)CCC(O)C(NC(=O)Cn2cnnn2)C1 c1(SCC(=O)NCC(CSC)OC)ccccc1.C12(CCSC1)C(=O)N2 N1(C(C2=NOC(CNC(C3(C#C)CCCC3)=O)C2)=O)CCN2CCOCC2C1 C(CC(C)CC)(C(=O)N1CCC12CCC2)NC(C(CCC)NC(N)=O)=O C(CCC(C)NC(c1n[nH]c(C2CC2)n1)=O)NC(CCOCCCOC)=O C(=O)(CC(C(C)CC)NC(C1COC(=O)N1C)=O)NC(CC#C)C(=O)OCC c1(C(N(CCCNC(C2(C)CC(F)C2)=O)C2CC2)=O)cncc2c(F)cccc12 Cc1[nH]c(=NCC=CCNC(c2occ3c2CCC3)=O)ccc1C#N N1(C(Cc2cc(C)nn2C)=O)CCOCC(C(=O)N(CC(F)(F)F)C)C1 c1(C(=O)NCCC(C)NC(CC(=O)OC)=O)ccc2c(c1)n(C)c(=O)n2C C1(OCC)CC2(C1)CC2C(=O)OCc1ccc(-n2cc(CCN(C)C)nn2)cc1 C1(CNC(c2ccc(Cl)nc2O)=O)CN(C(C2COC2)=O)C2CCN1C2 C1(C(=O)NCC(C(C)C)NC(CC(C=C)(C)C)=O)CC2(CC(C)=NO2)C1 N1(C(c2n(COC)ncc2)=O)CCCN(C(C2CCC(O)C2)=O)CC1C CCCCCCCCCOC(c1ccc(C(C)(C)C(F)(F)F)cc1)=O N1(C(C(C)C2CC2)=O)CCCC(N=c2c(Br)c[nH]cc2[N+](=O)[O-])CC1 C(=O)(CCC(C)NC(=O)C(C)(C)Cl)NC(CSC)C CON(C)CCCN=c1[nH]c(C)cc(=NCC2CC2Cc2ccccc2)[nH]1 c1(C(C(=O)NCCCSC)N(CC(C)C)CCC)ccc(F)c2c1CCC2 c1(-c2scc(C(N3CC(OC)C(C)CC3)=O)n2)cc(C(F)(F)F)ccc1Cl c1(C(C(=O)NC2C(NC(CCCCCCC)=O)CC2)C)cn(C)c2ccccc12 N1(C(C2(OC)CC2)=O)CCC(C2CCCN(C(=O)C3=C(Cl)CCOC3)C2)C1 C(=O)(CCC(=O)Nc1cccs1)NCC(C)(C1CC1)NC(CC=CCC)=O c1(CNC(CN(CCC)C)=O)ncoc1C1CN(C(=O)C(C)SC)C1 CC(F)(F)CC(=O)NCC1(C(C)(C)O)CN(C(=O)COCC2CCCOC2)C1 c1(C(N2C(CCCNC(C3C(OC)CC3)=O)CCCC2)=O)ccn2nccc2c1 C(=O)(C(C(C)C)NC(=O)COC(=O)C=Cc1ccsc1)NC(C1CCCC1)CC C1(CC)CCCCC1C(=O)NCC1(NC(c2cnn(CCF)c2)=O)CCOCC1 c1(C(N(C(CNC(c2cc(CCC)nn2C)=O)C)C)=O)ccc(C)cc1SC N1(C(C(C)(C)OCC)=O)CCN(C(=O)CC2CC(C(=O)OC)C2(C)C)C(CF)C1 N(C1CN(C(c2c(Cl)noc2C)=O)CCc2ccccc21)C(CC(C=C)C)=O N1(C(C=C2CCC(C)C2)=O)CCC(NC(c2conc2C(C)(C)C)=O)C(C)(C)C1 C1(CCC)(C(N2CC3C(c4cn(CCC(F)(F)CO)nn4)C3C2)=O)CCNC1=O c1(OC)cc(C)c(CN(C)C(C2CCCN2CC(C)C)=O)cc1NC(=O)C(F)(F)F N1(C(CCC2CCN(C(C3(CO)CC(C)C3)=O)C2)=O)CCN2CCCCC2C1 C12(C(=O)NCCCNC(c3c(C(=O)OC)ccs3)=O)CC3CC1(CO)CC3C2 C(=O)(C1CCOc2ccc(F)cc21)NC(c1cn(-c2c(C)cccc2)nn1)(C)C N1(CC)C(=O)CCC1C(=O)NCC1(O)CC(NC(=O)CC2CCC2)C1 CCC#CCCNC(C1C(C)CN1C(=O)CC1(O)CCOC1)=O Cc1cc(C)c(S(=O)(=O)NC2CCC(NC(c3sccc3F)=O)C2)c(C)c1 CCCCC(O)C(C)C(=O)N1CCN(C(c2cccc(C)n2)=O)CC1C CCC(C)CC(=O)C(=O)N1Cc2occ(C(N3CC(c4ccccn4)C3)=O)c2C1 Cc1cc(C(=O)NC(C2CCCN2C(=O)CSc2nc[nH]n2)(C)C)c(Cl)cc1F C(=O)(C(C)(C)CS(N)(=O)=O)NC1CC(C)(NC(=O)C(O)Cc2cccc(Cl)c2)C1 N1(CC)CC(Nc2ncnc(N(C)Cc3ccoc3)c2C)CCC1=O C1(C(N2C(C)(C(=O)NC)CC2)=O)CCC(C)(C)N(C(=O)C(C)CC#N)C1 c1(C(=O)NCC2C(CC(=O)NC(c3nc[nH]n3)CC)C2)cccnc1NC1CC1 c1(C(=O)NC2CCCCN(C(c3ccc(C#C)cn3)=O)C2)ccc(C)c(C#N)c1 C1(NC(CCCSC)=O)CCC2CN(C(=O)C(C3CCC3)OCCO)CCC2C1 c1(N(C(=O)C(F)OC(F)(F)F)Cc2ccc(C(C)C)cc2)cncc2cnccc12 C(=O)(C(C)CCCC(C)C)NCC(=C1CN(C(C(CCC)CC2CCCC2)=O)C1)F CC1CCN(C(c2ns[nH]c2=O)=O)CC1CNC(C1(CO)CCCCC1)=O CC(C(=O)N1CC(NC(c2cnc(O)c(Br)c2)=O)C2(CC2)C1)C(C)(C)C C1(CC=C)CCCCC1NC(c1cccc(CC)n1)=O.C12C(C1(C)C)C(=O)NC2 N1(C(C(CC(C)C)C)=O)CC(C)(C)OC2(C1)CN(C(c1cc3sccc3s1)=O)C2 CC12CCC1CN(C(=O)C(c1cccnc1)NC(=O)C(c1ccccc1)F)C2 c1(C(=O)OC)n[nH]c(C(c2ccnn2C)CC(=O)OCCC=CC)c1C C1(NC(=O)CNC(=O)Cc2ccco2)CCCN(C(=O)CCOC(F)F)CC1F C1(O)(CNC(C(C(C)NC(c2ccc(CF)cc2)=O)C)=O)CCCCCC1 c1(C(=O)NCc2ccc(CNC(c3cnc(C)s3)=O)cc2)cncc(N)c1C c1(C(N(CCNC(=O)Cc2cc(O)nc(O)n2)CC)=O)ccccc1S(=O)CC C=CC(C)(CC)C(=O)NCC1(O)CC(CNC(c2cnnn2C2CC2)=O)C1 c1(C(N(C)CC2CCN(C(=O)CCc3ccoc3)C2)=O)cnc(Cl)c(N)c1 C1(C(=O)Nc2ccc(OC)nc2C)CCCN1NC(=O)C12CCC(OC)C1C2 C(N=c1[nH]c(C#N)c(Cl)s1)C1CN(C(C2CCC(OC)C2)=O)C1 c1(C(=O)NCC2(CNC(C(C(=O)OCC)CC)=O)CCC2)ccc(S(C)=O)cc1 C1(NC(C=CC(=O)OCCCC)=O)CC(C)N(C(c2n[nH]c(C)c2Br)=O)C1 C1(NC(CSCC=C)=O)CCCN(C(c2cc(OC)cc(Br)n2)=O)C1C c1(C(=O)NC2C(OC)CN(C(=O)CSC)C2)ccc(C)c2cccnc12 c1(CC(=O)NC(c2ccc(CNC(CC(CC)O)=O)cc2)C)cc(O)nc(O)n1 C1(C#N)(C(=O)NCC2C(C(N(C3CC4CCC3O4)C)=O)C2)CCOC1 c1(NC(c2c(Nc3nc(C)cc(SC)n3)c[nH]n2)=O)nc(Cl)ccc1C#N C=C=CCCC(=O)N1CC(OCCNC(=O)CSc2ccc(F)cc2)C1 C1(C)(CNC(c2cnc(CCC)s2)=O)CN(C(C2CC(C)(O)C2)=O)CC1C c1(CS(Oc2ccc(CC(=O)OC)cc2)(=O)=O)ccc2ocnc2n1 c1(C(N2CCC(NC(C=CCN(C)CC)=O)C(F)C2)=O)c(F)ccc2ccoc12 C1(C(=O)NCCSC)(NC(c2ccc(Cl)cc2O)=O)CCC(n2ccnn2)CC1 Cc1nc(C(=O)N(C(C)CNC(=O)C(c2cccc(Br)c2)(C)C)C)c(C)o1 c1(C(N2C(CNC(c3c(C)nccn3)=O)CCC2)=O)ccc(CO)c([N+](=O)[O-])c1 Cc1ncc(Cl)cc1C(=O)NCC(CNC(C1COCCN1C)=O)CO CCC(C)(CC(=O)NC(c1ccc(F)cc1F)CNC(=O)CN(C)C)C(=O)OC N1(C(C(C)OCCN(C)C)=O)CC(C2CCCN(C(C3(C)CCC(=O)N3)=O)C2)C1 C1(C(=O)OC)CN(Cc2nc(C)cn2C)CC12CC2 N1(C(C(C(=O)OCC)F)=O)CC(CNC(c2nn[nH]c2C(F)(F)F)=O)CC1(C)C c1(SCC(=O)NCc2cn(CC3CCCO3)nn2)ccccc1C(F)(F)F C1(CN(C(c2c(CC)c[nH]n2)=O)C)CN(C(=O)C=CC2CCCO2)CCO1 c1(C(F)(F)F)n[nH]c(=NC2CC3OC(C(F)(F)F)COC23)s1 C(=O)(CCC(F)F)NCCC(C)N(C)C(c1cc(Br)n(C)c1)=O c1(CNC(CC(C)F)=O)cccc2c1CN(C(c1cccc(O)n1)=O)C2 C1(CNC(=O)NCC(CC)(C)c2ccccn2)CN(C)CCN(C)C1 CON(CCC(=O)NCCn1cnc(CO)c1)C(=O)C1(C)CC(C)C1 c1(OC)ccc2cc(C(=O)NCC34CC(CN3C(C3(SC)CC3)=O)C4)sc2c1 Cc1ncc(C(=O)NCCC2(O)CCCN(C(c3nnsc3C)=O)C2)cc1Cl Cc1cc2n(n1)CCN(C(C1CN(C(c3n[nH]c(=N)[nH]3)=O)CCN1C)=O)C2 Cc1ccc(CC(=O)NCCC(C)NC(=O)C(F)(F)c2cnn(C)c2)cc1 C(C(C)C(C)C(=O)NCCN(C(=O)CCc1ccon1)C1CCCC1)OC Cc1csc(=NCC(=O)N2CCC3CCN(C(=O)CCS(=O)(=O)N(C)C)C3C2)[nH]1 c1(C(=O)NC(C=CCNC(CN2C(C)CC2)=O)(C)C)cc(C2CCC2)nn1C C(=O)(C(C)CC(=O)c1ccccc1F)NCC1(O)CN(C(c2c(C)nsc2)=O)C1 N1(C(C(CSC)C)=O)CCC2OCCN(C(c3cc4cccnn4n3)=O)C2C1 C1(CNC(=O)C=C(Cl)Cl)CC2COCC2N1C(=O)CN1C(=O)CNC1=O C(=O)(C1=CC2C=CC1C2)NC1CCCC(C(N(CC(=O)OCC)C2CC2)=O)C1 CN1CC(NC(c2ccoc2C2CC2)=O)C(c2ccccc2)C1 c1(C(=O)NC2C(NC(C3CC(C(=O)OC)C3)=O)COCC2)c(F)ccc(C)c1F c1(SC)cccc(C(=O)NC(C)(C)CCNC(c2cc(Cl)nnc2O)=O)c1Cl c1(C(N=c2[nH]n(CC(CC)OC)c(C)c2)=O)cc2[nH]nnc2cc1OC C1(NC(C2CC3(CCO2)CC3)=O)CN(C(c2cc(Cl)ns2)=O)CCC12CCC2 N1(C(C=CC=CC)=O)CCCCC1CCC(C)(C)NC(c1csc(C)n1)=O c1(C(=O)NCC(C)(C2CC2)NC(c2ccsc2)=O)ccc(Cl)c(F)c1 C1(C(NOCC#C)=O)CCC(C)(C)N(C(=O)COCCN(C)C)C1 CC(C)C(CCC(F)F)NC(=O)NC1CC(C)(C(C)(C)C)C1 c1(C(=O)NC(C(C)NC(c2cc(N)cc(O)c2)=O)C)cc2c(F)ccc(F)c2[nH]1 C1(NC(C(c2cccc(O)c2)C)=O)CC12CCN(C(=O)C(C)(C)N(C)C)CC2 c1(C(=O)NC2C(NC(C(CC=C)(F)F)=O)CCC2)ccc2c(c1)CCCC(=O)N2 c1(C(N2CC(OCCNC(C3C(OCC)CC3)=O)C2)=O)ccc(C(F)F)nc1O c1(CC)c(OC)cccc1C(N1CCN(C(=O)CCCF)C(CCO)C1)=O c1(OCCOC)cccc(NC(c2nc(C)c(Br)s2)c2nnnn2C(C)C)c1 c1(N2CCCC(C(C)NC(c3cccc(OC)c3Cl)=O)C2)nc(C)ncc1C#N C1(C(N(C)Cc2c(CNC(CC3CC(C)C3)=O)cccc2)=O)CCC=CCCC1 c1(SC)cc(O)ccc1NC(c1ncc(Cl)n1C)c1nnnn1C1COC1 N1(C(C(CC)F)=O)CC2(CC2)CC1CNC(=O)C(c1ccccc1F)(C)C C1(C(C)(C)NC(c2c[nH]nc2C2CCCO2)=O)CCN(C(=O)Cc2ccon2)CC1 C#CC1(C(=O)NCC2CCC(C(=O)NC(C)C(O)C(F)F)C2)CCCC1 C(=O)(C1=CCCSC1)NC1CC(CNC(CCCCN(C)C)=O)C1 N1(C(C2(CC)CC2(F)F)=O)CCC(O)(CNC(c2cncc(O)c2)=O)C1 C(CNC(=O)C(Cl)=CCl)(C(C)C(C)C)NC(c1c(CSCC)cccc1)=O C1(NC(c2cc(CCNC(CC)=O)on2)=O)CC(CO)N(C)C1 C1(NC(c2c(C)oc(-c3cccs3)n2)=O)CCCCN(C(=O)C(C)C#N)CC1 N(C1CCc2c(Cl)cc(Cl)cc21)C(C)C(C)Sc1ccccc1 CC1CC(NC(C2CCC2NC(c2cc(O)ncc2F)=O)=O)CC(C)(C)C1 Cc1c(CS(=O)(=O)Cc2ccc(F)cc2)noc1-c1ccccc1OC(F)F N1(C(C2(OC)CC2)=O)CC2CCN(C(=O)C3CC3)CC12.c12ncc(s1)n2C Cc1cc(=NCc2ccc(-c3cccs3)o2)[nH]c(NC(c2cccc(Cl)c2)C)n1 C(C(C)(C)C(C)(F)F)NC(C=CCC1(NC(C(CC)N(C)C)=O)CCC1)=O C1(C(=O)NCC(C(=O)N(CCCC#C)C)OC)CC12CCOCC2 C(=O)(CCSC)NCCN(CCOC)C(C1CC1(Cl)Cl)=O C(=O)(C1=NOC(C)C1C)N1CCC(C(=O)Nc2ccccc2O)(OC)C1 C(=O)(C(C)(C)C(C)(C)O)NCC(C)(C1CC1)NC(C(CC1CCC1)OC)=O Cc1ccc(C(C)NC(=O)CC(c2cccc(C(=O)O)c2)C)cc1Cl N1(C(C(CC=CC)C)=O)CC2(CC(C(=O)N(C3CC(CO)C3)C)CO2)C1 N1(CCN=C(NCC2(C(=O)OC)COC2)NCC(F)F)CCCC(C)(C)CC1 NS(=O)(=O)c1ccc(C(=O)NC2C=CCN(C(=O)Cc3ccoc3)C2)cc1 CN1CC=CCC1CC(=O)NC1CC2(C1)CC2NC(=O)CC1CC2(CCC2)C1 O=C(C1=CCCOCC1)NCCCCCNC(C1CCC2(C1)CC2(F)F)=O C=C1CC(CC(=O)N(CCN(C)C(C2CC2(C)C(C)C)=O)C(C)C)C1 C(=O)(C(C)S(=O)(=O)C(C)C)N1C2CC(CNC(c3c(C)nc(C)n3O)=O)C1CC2 c1(CCC)cc(N(C2CC(C(=O)OCC)C2)C=O)ncn1 Cc1cc(Br)cnc1C(=O)N(c1ncc(F)c(C)n1)CCCN1CCNCC1 c1(C(c2n(C(CC)C)nnn2)NCc2ccncn2)cc2ccccc2s1 C1(NC(c2ncc(Cl)cc2F)=O)CN(C(=O)C2=CCCOC2)CC12CCOCC2 CC1CCCC=C1C(=O)N1CC(C)(NC(C2CC(O)C2)=O)C1 N1(C(CC2CC(C)(C)OC2)=O)CCC2CCC(C1)N2C(C12CC(C1)C2)=O N1(C(Cn2c(C)nc(C)n2)=O)C(C(=O)NCC(C)C2CCC2)CCC12CC2 C1(C(=O)NCC(C)CC2CCC2)(NC(COC)=O)CCC(C)(C)C1 c1(CC(C)(C)CO)nc(C2CN(C3CCOC3)C2)n(C2CCCSC2)n1 N12CCC(C1)SC1(CC1)C2=O.c1(COC(C2CCOC2)=O)ccccc1 c1(C(N(C2CN(C(CCCC#C)=O)C2)C)=O)ccc(OC(F)F)cc1F CC(CN=c1[nH]c(N2CCOC3(CC3)C2)nc2c1SCC2)C(F)(F)F.CC Cn1nnnc1C(C)(CC1CC12CCC2)NC1CC(C2CC2(Cl)Cl)C1 C1(O)(C(C)NC(Cn2c(C)ccn2)=O)CCN(C(=O)C(C)CCO)CC1 N1(C(C(CC=CC)C)=O)CC2(CNC(=O)C#CC3CC3)CCC1C2 N1(C(c2cc(N)c(Cl)cn2)=O)CCC2(CC1)CC(NC(c1ccco1)=O)CCO2 Cn1nc(C(F)F)c(CNC2CC(F)CN(C(c3ccncc3Cl)=O)C2)c1Cl c1(CN(C(=O)NC2(C)CCC(C)C2)C)cc(Cl)cc(Cl)c1 Cc1c(CC(=O)NC2CC(F)(Cc3cn(CCF)nn3)C2)oc2ccccc12 N1(C(C2(CC#C)CCCO2)=O)C2CCC1CN(C(C1CC1C1CC1C)=O)C2 C1(C(N(CCNC(=O)CCN2CCCCC2)C2CC2)=O)C(Cl)(Cl)C12CC2 C1(NC(C2CCCN(CC)C2)=O)(CO)CCN(C(C2CCCC2CF)=O)CC1 c1(C(=O)NC(CCC)CNC(=O)CNC(C2CC2C)=O)cn(C)c(C)n1 c1(OC)nccc2c(C(=O)NCCC(C)NC(C3CCC4(CCC4)O3)=O)c[nH]c12 C1(NC(=O)CCCc2cc[nH]n2)COC2(CCN(C(=O)CSC(F)F)C2)C1 c1(CCC(=O)N(C(C)CO)CCC)cc2ccc(O)cc2oc1=O C#Cc1ccc(C(N2CC(NC(c3cc(Br)ccc3F)=O)C3CC23)=O)cn1 N1(C(C(C)(C(C)C)OC)=O)CCC2(CCCN2C(c2csc(F)c2)=O)C1 C1(CNC(C2CC(CCC)C2)=O)COCCN1C(=O)CCCc1ncc(C)o1 Cc1cc(C(N2CC(NC(=O)CCCc3cccs3)C(F)C2)=O)oc1C N1(C(C2N(CC)CCC2)=O)CCC(C2(NC(=O)CCc3cnn(C)c3C)CC2)C1 Cc1cc(N2CCC(CNC(c3cccn3Cc3cccs3)=O)CC2)nc(Cl)n1 c1(CN(C(=O)C(CNC(=O)C(C)(C)C(C)C)OC)CC)ccc(F)c(F)c1 C1(CC)CCOCCN1C(C1N(C(=O)C(C)COC(C)=O)CCC1(C)C)=O C1(CNC(=O)Nc2cccc(C(F)(F)F)c2)(NC2CCS(=O)(=O)C2)CCCCC1 C1(CC(=O)N(CCC(=O)NCCC2(C)CCCC2)CC)CCC(C)(C)C1 N1(C(c2nc(CC)oc2)=O)CC2CCC(C1)N2C(c1ccc(Cl)c(Cl)c1N)=O C(=O)(CC(O)CNC(C1CCC=CCC1)=O)NC1(C)CCOC1 CC(C)(O)CC(C(=O)Nc1ccc(-c2nn[nH]n2)s1)NC(=O)OC(C)(C)C C=C1CCC(C(=O)NC2CN(C(=O)Cc3cc[nH]c3)CC2n2cccn2)CC1 CCC(C(=O)N1CCN(C(=O)CN2CCCCC2)CC1)C(C)O N1(C(CCNC(C)=O)=O)CCC(C)(C)C(CNC(=O)CC2C=CCCC2)C1 N1(C(CNC(N)=O)=O)CC(NC(C2CC2F)=O)C2(CCS(=O)(=O)CC2)C1 c1(C(N2CCC(NC(c3c(CC)ncs3)=O)C(F)C2)=O)ccc(F)c(C#N)c1 CC1CCC(N=c2[nH]c3ccc(S(=O)(=O)NCCCCCCO)cc3s2)C1 c1(C(N2CC=CC2Cn2cc(CC3(n4nccn4)CC3)nn2)=O)ccc(F)c(F)c1 n1(CC)c(C)cc(C(=O)NC2CC2NC(c2cnc(C)nc2C)=O)c1C c1(C(N2CC=CC(C(N(C)CCOC(F)F)=O)C2)=O)nccc2[nH]ccc12 C1(C)(COC)CCN(C(c2cc(CNC(C3CCOCC3)=O)cs2)=O)CC1 c1(SCC(=O)N(C)CCN(C)C(c2cnoc2C2CCC2)=O)ccccc1Cl N1(C(CN(C(COC)=O)C)=O)CC2CC2(CNC(C23CC(C)C2C3)=O)C1 c1(N2CC(CC=C)(NC(=O)C3=CCCC3)C2)cc(C)nc2c(C)cnn12 N1(C(C2CC23CCC3)C(=O)NCC(C)C)Cc2cncnc2C1 c1(C(C(=O)NCCN(C(C2SCCS2)=O)CC)OC(C)(C)C)ccccc1 N1(C(C(CC=C)(C)C)=O)CCC2(C1)CN(C(c1ncc(Cl)nc1Cl)=O)CCO2 c1(C(N2CCCC(C(C)(C)C(=O)NCC#CC#CCO)C2)=O)ccc(O)c(F)c1 c1(CNC(CC=C)C(=O)N2CCOCC2)cc(Cl)cc(C)c1[N+](=O)[O-] CON(C)C(=O)CN=c1cc(C)[nH]c(=NC(C)C2CCCO2)[nH]1 c1(C(=O)NCCC(CNC(C(C2CCCC2)OC)=O)O)cc(C)n(C2CC2)n1 C1(NC(CC2C(CC)C2)=O)CCCCC1CC(=O)Nc1csnc1C CC(C)C1=NOC(C)(C(N2CCN(C(C3CCNC(=O)C3)=O)C(CO)C2)=O)C1 C1(CC(=O)NCC(C)(C)NC(C(CC)NC(N)=O)=O)CCCC2(CC2)C1 C(C(C)CC(=O)N1CC2C(NC(c3[nH][nH]c(=N)c3Br)=O)C2C1)OC c1(C(=O)NCCN2CCN(C(C3C(OCC)C3)=O)CC2)ccnc(Cl)c1N c1(CC(=O)NC2C(NC(C3=CC(C)(CC)C3)=O)CCC2)c(N)nc(C)nc1O n1(CCCC(=O)N(CC(F)F)C)c(=O)oc2cc([N+](=O)[O-])ccc12 N1(C(C2N(C)CCC2)=O)CC2CCC(N(C(=O)C=CCn3cncn3)C)C2C1 c1(C(=O)NCC(=O)Nc2ccccc2)ccc2nn[nH]c2n1 Cc1ccncc1CC(=O)NC1COCC1NC(C1(C2CCCO2)CCCC1)=O C(=O)(C1=Cc2ccccc2C1O)N1CCC(NC(Cc2c(C)non2)=O)C1C c1(CC(N2CC(C(C)NC(C3CC3c3ccoc3)=O)C2)=O)ccc(F)cc1F Cc1ccccc1-c1nc(CN2CCC(N3CC(C)(C)C3=O)CC2)c(C)o1 C1(C(N2CC(F)(CNC(C3C(C#C)C3)=O)C2)=O)Cc2cc(C)ccc2S1(=O)=O N1(C(C2(CC#C)CC=CCC2)=O)CCCC(C2CN(C(C3(C(C)=O)CC3)=O)C2)C1 C1(C(N2CCC(CC#N)CC2)=O)CN(C(=O)CSC(F)F)CCCO1 c1(C(N(CCCCCNC(CSCCC)=O)C)=O)cc2c(cc1Cl)OCCO2 N1(C(C(CC)CC)=O)CCC2(CC1)CC(NC(=O)CN(C)S(N)(=O)=O)CCO2 C1(NCc2c(C)nn(-c3ccccc3)c2C)Cc2cnccc2NC1=O C(N=c1cc(NCC2(C(F)(F)F)CCC2)nc[nH]1)C1(C)CCC(F)(F)C1 N1(C(C)C)CCN(CCC2CCCC(F)(F)C2)CC1=O N1(C(c2c(C)nco2)=O)CC2CCOCC2(NC(c2ccc(C(C)C)cc2)=O)C1 c1(C(=O)NC(CNC(C(C(CC)O)C)=O)CC(C)C)ccc2cnnc(O)c2c1 Cc1nc(C(C)NCc2ccc(OC(F)F)o2)c(C)o1 c1(C(N(C2CCN(C(=O)CCC3CC3)C2)CCC)=O)oc(CCOC)nc1C C1(C(N(CCn2cc(CC(O)C(C)C)nn2)CC)=O)CCC(C)(C)OC1 N1(C(C=COCC)=O)CCCCC1C1(C(=O)NC2CC(C)(C)CO2)CC1 Cc1cc(C#N)cnc1C(=O)NC1CCC(C)N(C(=O)C=Cc2cnc[nH]2)C1 Cc1noc(C(C)C)c1C(N1CCN(C(C2CCOC2=O)=O)CC1)=O c1(C(=O)NCC2CN(C(c3c(C(C)C)cco3)=O)C2)nnn(C2CCOC2)c1C c1(CC)csc(CNC(c2nnnn2C2CCCC2)C2CC=CCC2)n1 Cc1cc(F)ncc1C(N1CCC(CF)(NC(=O)CCCc2cccs2)C1)=O Cc1nccc(C(=O)NCCN(C)C(C2CC3(CCCC3)C2)=O)c1N N1(C(c2c(C)nc[nH]2)=O)CCOCC(NC(c2cc(CO)on2)=O)C1 C(CCC[Si](C)(C)C)N(C(c1ccc(SCC2NC(=O)NC2=O)cc1)=O)CC C#CCC(C)(C(=O)NC(C)(C)C#CCC)NC(c1ccoc1Cl)=O N1(C(C(C(=C)Cl)(C)C)=O)CCC2(CC1)CCN(C(c1cc(=O)n(C)cn1)=O)C2 C(CC(C)(C)C(=O)N1CCOC(C(C)(C)C)CC1)NC(CC1(N(C)C)CCC1)=O c1(C(C)(F)F)ccccc1C(=O)NCC1CCCCN1C(C1CC1C(F)F)=O C=C1CCN(C(c2cc(O)ncc2F)=O)C(C(N2CCC(CC)C2CC)=O)C1 Cc1c(C(=O)NCC2CCC(NC(=O)C=CC(C)C)CC2)oc2ccccc12 C1(C(=O)N(C)CC2CCOC2)(NC(CN(CCOC)C)=O)CCN(C)C1 c1(C(=O)NC2CCCC(NC(c3cccc(C)c3F)=O)C2)cc2cccnc2[nH]1 CC(C)CC(O)CC(=O)NC1CN(C(C2CCC(=O)N2C2CC2)=O)C2CCCC12 c1(C(C)NC(C2C3CCC23C(C)OC)OC)cc2n(n1)CCCC2 C(=O)(C(F)(F)C(O)C1CC1)NC(CNC(c1c(CC)non1)=O)C c1(CC)ccc([N+](=O)[O-])c(C#N)c1.C1(Cc2n(C(C)C)nnn2)CC(S)C12CCC2 C(=O)(C(C(=O)NC)OC)N(CCCn1cc(CCSC)nn1)CC c1(C(N(C(C)C)CCN(C)C(C2(O)CCC2)=O)=O)cc2ccccn2c1 N1(C(CC(=O)N(C)C)=O)CCN(C(c2ccc(I)cc2)=O)CC1 CC1CC(NC(=O)Cn2ccnn2)CCN1C(=O)C(=O)C(C)(C)C CC1CC=C(C(=O)N2CC3CCC(CNC(C4CCCC(CO)O4)=O)(C3)C2)CC1 c1(CC)cncc(C(=O)NC2(CCC(=O)NCC3CCN3CC)CCCC2)c1 C(=O)(CC(C)C(C)(C)C)NC(CCCC)CNC(=O)C(=Cc1cccs1)C c1(OC)cccc2c1OCC(C(=O)NCC(C(C)C)NC(C1(C)CSC1)=O)C2 c1(N2Cc3c(nc(=N)[nH]c3)C2)nc2c(c(=NC3CCCc4[nH]ccc43)[nH]1)CCC2 CN1CC(C)(C)CC1C(=O)NC1CCOCC1NC(=O)CSc1nncn1C CCC(CC)(CO)C(=O)NCC1C=CCN1C(=O)CCCSc1ccccc1 N1(C(Cc2cnc(C)[nH]2)=O)CCC2CCN(C(=O)Cc3cccc(C)c3C)C2C1 C1(CCCC)(C(=O)NCC(CO)NC(=O)Cn2cnnc2O)CCCC1 c1(C(N(CCNC(=O)C=Cc2ccccc2)CC)=O)ccc(Cl)c(C(F)F)c1 C=CCC(CNC(=O)CC1(OCC)CCC1)NC(=O)Cc1nncn1C(C)C C(C(C)(C)C(=O)NCCCCCN(C(=O)CC1CC2(CC2)CO1)C)N(C)C C1(C(=O)NC(c2ccc(C)o2)Cn2ccnc2)C2C=CC(CC2)C1C(=O)O C#Cc1ccc(C(=O)NCC2(CNC(C3CN(C(C)C)C3)=O)CCCC2)cc1C c1(CN(C(C(CCC)O)=O)CC)c(C)cc(C)c(C(=O)O)c1C CC1CCC(C(=O)NC2(CN(C)C(c3cnns3)=O)CC2)C(=O)N1 c1(CC)cc([N+](=O)[O-])ccc1C(=O)N(CC(C)NC(c1ccc(Cl)c(Cl)c1)=O)C c1(C(N2CCC(C(=O)NC(C3CCC3)C)C2)=O)ccc(OC(F)F)cc1 N1(C(c2c(C)ncnc2)=O)CC(CNC(=O)C(C)(C)C2(C)CC2(F)F)C2(CC2)C1 C1(CC(=O)N(C)CCn2ccnc2)C2CCCC2N1C(c1ccc([N+](=O)[O-])o1)=O C(=O)(CC1=NNC(=O)C1)NCCC(=C)CNC(C1(C)CCCC1(F)F)=O C1(O)(CN(C(=O)CCC(F)F)C)CCN(C(=O)CCCC2CCOCC2)C1 N1(C(C2(CNC(c3c(C)oc(Cl)n3)=O)CC=CC2)=O)CC2CC(C)C2C1 N1(C(CCC)=O)CCC2(CCC2)C(CNC(C2(CO)CCCO2)=O)C1 Cc1nc(C)c(C(N2CC3(CC3C(=O)Nc3cscn3)C2)=O)[nH]1 C12(NCCN(c3ccc(F)cc3)C(c3c(C(C)C)ocn3)=O)CCC(C1)OC2C c1(OCCC(N2CC(CNC(CCC=C=C)=O)OCC2)=O)ccc(Cl)c(F)c1 CC(CCC(=O)NC1CC(CCF)C1)NC(C1CCC2CC12)=O c1(NC(c2nc(C(=O)Nc3cncc(C)c3)sc2)=O)ccc([N+](=O)[O-])cc1C N1(C(CC(CC)C2CC2)=O)CCC(C2(NC(C3CCOC3C)=O)CC2)CC1 c1(OC)cncc(C(N2CC(N(C)C(c3ccn(C)c3)=O)C2)=O)c1 C(=O)(NNc1c(Cl)cc([N+](=O)[O-])cc1Cl)NC1CN(C(C)C)C(=O)CC1 C1(CC)CN(C)C(=O)CN1C(=O)C(CC(F)F)NC(C1CCC1(F)F)=O C1(CNC(C(C)O)=O)(CNC(c2cc(CS(C)(=O)=O)on2)=O)CCCCC1 C1(C)(CC)CCC(NC(=O)CN(C)C(c2cccn(C)c2=O)=O)CC1 N1(C(C2(OC)CCC(C)(C)C2)=O)CCC2CCC(C1)N2C(c1csnn1)=O c1(OC)cc(Br)cc(F)c1CN1CCC(CC(=O)Nc2scc(O)c2C#N)C1 C1(CCNC(CCCOCC=C)=O)C(C)CCCN1C(c1cc(=O)n(C)cn1)=O c1(CCC(N2CCCCC(NC(=O)CSC(F)F)C2)=O)ccc2ncsc2c1 c1(C(=O)NCC2COCCN2C(C2(Br)CCC2)=O)cnc2ccc(Cl)cn12 C(=O)(CC(C)CC(=O)OC)N(CCCNC(=O)C=CCO)CC C1(NC(C23C(C)(C)OCC2C3)=O)CC2CCC1CN(C(=O)Cc1c[nH]nc1O)C2 c1(CC)nc(C)oc1C(N1CCC(CNC(c2cn(C)nc2OC)=O)(OC)C1)=O C1(C#N)(C(N(CCC2CCN(C(C3(OC)CCSC3)=O)CC2)C)=O)CCCCC1 c1(CCC(=O)NC(C)CNC(=O)C(c2ccnn2C)O)ccc(Cl)cc1 C(CNC(=O)C(c1cccc(Cl)c1)O)(CC(F)(F)F)NC(c1cc(C)c(C)[nH]1)=O C1(C(=O)NCCC2CCCN(CC(=O)NCCC(C)(C)C)C2)CCCC(F)(F)C1 C1(C(=O)NCC2C(C)CC2)(NC(=O)CC2CSCCO2)CC(F)(F)C1 c1(C(N2C(C)CCC(NC(C34CCN(CC3)C4)=O)C2)=O)ccc2nncn2c1 c1(CNC(C(=O)NCc2cc(C(C)(C)C)no2)=O)ccc(Cl)cc1F c1(NC2CCC(CNC(c3ccon3)=O)C2)cc(OC(F)F)ccc1[N+](=O)[O-] N1(C(=O)CCOc2cccnc2)CCC2(CCCN2C(C2CC(O)C(F)C2)=O)C1 C(=O)(C(C)(O)c1ccccc1)NC(CN(C(=O)C(O)CSC)CC)C c1(C(=O)NCCC2(CNC(=O)CC3C=CCC3)CC2)cc2c(=O)[nH]ccn2c1 C1(C(N2CCCC(C=C)C2)=O)CN(C(c2c(C)cncc2C)=O)CCC1(C)C Cc1cc(C(F)F)oc1C(=O)NC1(CNC(=O)C(C)(C)n2cnnn2)CCC1 CC(C1CCCCC1)=CC(=O)NCCC(C)(C)NC(c1cnc(CC(C)C)s1)=O C=C(C)CC(C)C(=O)NCC1CC1NC(c1ccc(OC2CC2)cc1)=O C1(CC(=O)N(C)CC2COCCN2C(=O)Cn2ccc(=N)[nH]2)CCC(C)(C)CO1 N1(C(Cc2cc(C)on2)=O)CCCC12CCCN(C(c1n[nH]cc1C1CC1)=O)C2 N1(C(c2ccc(CN=[N+]=[N-])o2)=O)CC=C(CNC(c2ccnnc2Cl)=O)CC1 Cn1cc([N+](=O)[O-])c(=NCC2CN(C(=O)CC3COC(=O)C3)CC2(C)C)[nH]1 CCC(C)C(c1ccccc1)NCCCn1nnnc1O C(CO)(C(C)(C)CO)NC(N(C1CCCN(Cc2ccccc2)C1)C)=O c1(OC)cccc(NC(=O)C(C2(O)CCC2)NC(=O)CC(C)SC)c1 CC(CCC(C)(C)C)C(=O)NCC1CCC2(CN(C(c3ccc(C#N)s3)=O)C2)O1 c1(SCC(=O)NCCC(C)NC(C(C)c2ccsn2)=O)ccc(Cl)cc1 N1(C(C(C=CC)O)=O)CC(NC(=O)C(C)(C)N2CCOCC2)C(O)C1 c1(OC)ccnc(CCC(N2CCOC(C(N3CCC3CO)=O)C2)=O)c1 C(C)(C(=O)NCC(C)(C)C1CC1)N(C(=O)COC(C)=O)CCC N1(CC(N2C(CNC(C3CC(OC)C3)=O)C(C)CC2)=O)CCCCCCC1=O N1(C(C2(CCC=C)CN(C(=O)C(C)CC(N)=O)C2)=O)CC(F)(F)CC1CO C#Cc1ccc(CC(N2CCN(C(C3CN(C)C3)=O)C(C3CCC3)C2)=O)cc1 CC(=O)C(C)CC(C)C(=O)N1CC(F)CC1C(=O)NCC(C1CC(C)(C)C1)O CCCS(=O)(=O)CC(=O)N1CC2CC1CN2C(=O)C(n1ccc(C2CC2)n1)C C1(NC(C2C(C)CCC2)=O)C2CCC1CN(C(=O)CCn1cnc(=N)[nH]1)C2 C1(CC(N)=O)(NC(CS(=O)(=O)NCC)=O)CCN(C(=O)COCC(F)F)CC1 C1(NC(=O)C(F)CC2CCC2)CN(C(c2cc(C3CC3)no2)=O)CC1C(F)F N1(C(c2cn(CCCC)nc2C)=O)CC2CCCC1CN(C(=O)COCCF)C2 C1(OCC)CN(C(C2(CF)CCOCC2)=O)CC1CNC(C1(CO)CCCC1)=O C1(OC(CC)=O)C(C)CCCN1C(=O)CSc1ccc(C(C)(C)C)cc1 N1(C(c2nc(C)c(C)s2)=O)CCC2C(NC(C3CCOC(C)C3)=O)C2C1 c1(C(N(C)CC2CCN(C(c3cc(C(=O)OC)[nH]c3)=O)C2)=O)n[nH]c(SC)c1Cl c1(C(N2CCC(COC)(NC(c3ncoc3C)=O)C2)=O)cc(SC)ccc1O C1(C(=O)NCCc2ncn(C)n2)(COC)CN(C(c2c[nH]cc2C)=O)C1 c1(C(=O)NCC(CNC(Cn2cc(C(=O)OCC)nn2)=O)C)ncc(C)cc1F c1(C(=O)NC23CCC(CN(C(c4cn(C)nc4)=O)C2)C3)ncccc1S(C)(=O)=O N1(C(C2(C(=O)NC)CC2)=O)CCN2CCOCC2(CNC(=O)C2=CCCCO2)C1 C1(CNC2(c3nnnn3C)CC(C)C2)CC12CC(OCC)C2.C(C)(C)(C)O C=CCCCCC(=O)N1CCC(C)(C)C1CC(=O)NC1CCCCC1CC C1(CC(=O)NC(C=C)(C)CC)CC(C)(C)CN1C(c1sc(O)nc1C)=O c1(C(=O)NC(C)(C)CNC(=O)CSCC2CCCCO2)cccc2ccsc12 N1(CCNC(C(F)NC(C)=O)=O)CCCN(C(=O)CC2CCN(S(C)(=O)=O)C2)CC1 c1(C(C)C)ccc(Cl)c(NC(=O)C(=O)NCc2ccsc2)c1 CC(C)CCC(F)C(=O)N(CC(O)CN(C(=O)C(F)(F)C(C)(C)O)C)C CCC(C(=O)N1CCC(NC(=O)C(c2ccccc2)N(C)CC)C1C)C(C)C N1(C(c2c(OC)nccc2)=O)CC(NC(=O)Cc2sccc2C)CC1(C)C C(C)(C(=O)NC1CC(CNC(=O)Cc2ccccc2Br)C1)(C(C)C)OC C1(NC(C(C(C)C)NS(C)(=O)=O)=O)CCN(C(c2cnn(CCF)c2)=O)C(C)C1 C1(C(N(CC)CC2CCN(C(=O)CNC(=O)C3CC3)CC2)=O)CCN(C)C(=O)C1 c1(C(=O)NCC(CC)NC(=O)COCc2ccncc2)cc2cc(C)ccc2[nH]1 C1(n2cc(C(CC)(C)O)nn2)CC2CCC(C1)N2C(=O)CSC1CCCCC1 CCC(C)(C(=O)NCCCOCCCNC(=O)C(CCOC)C1CCC1)OC c1(C(=O)NCC(CC)NC(=O)C#CC(C)(C)O)c(C)nn2cc[nH]c(=O)c12 C=CCCN=C(NCC(C1CCCCC1)O)N1CCCC(CO)(CO)C1 C(C1CCCC1)=C(C)C(=O)N(CC(O)CNC(C1CCCN1c1nccs1)=O)C n1(CCC(C)C)cc(CNC(=O)C(=O)NC2COCC2Cc2cc(F)n[nH]2)nn1 Cc1c(C(=O)NCCCCNC(=O)CC2COC(CN)C2)nn2c1CCCC2 c1(CC)ccc(-c2nnco2)c(C(=O)O)c1.N12CC(C(OC)C1)OCC2=O CC(CC(F)F)C(=O)N1CCC(C)(C)C1CNC(=O)Cc1cnoc1 c1(C(N2CC(C=C)C(NC(=O)C(CC(C)C)OC)C2)=O)cn2cc(Cl)cnc2n1 c1(NC(C23CC(C(N(CC=C)CC=C)=O)(C2)C3)=O)c(Cl)c(F)nc(F)c1Cl c1(C(=O)NCC2(O)CCCN(C(COCC)=O)C2)ccnc2c(Cl)c(C)ccc12 N1(CC)CCC(NC(=O)CCOCCN(C(=O)Cc2ccc(O)cn2)C)CC1 N1(C(Cc2ccc(C)c(O)c2)=O)CC(C)C(NC(=O)C=Cc2cccs2)C(C)C1 N1(C(C2C(c3cccc(C(C)C)c3)C2)=O)CC(NC(=O)C(C)(C)C#N)CCC1C Cc1ncnc(N2CC3CC(NC(=O)CC(C)(F)F)CC3C2)c1C#N c1(C(N2CC(C(=O)Nc3cnc(F)c(Br)c3)NCC2)=O)cc2ncccc2[nH]1 c1(NC(=O)NC(c2c(C)cc(F)cc2)CCC(F)(F)F)ccccc1S(C)=O C(=O)(CCC(=O)NC1(CNC(=O)C(c2ccccc2Cl)OC)CC1)NCC n1(C2(C)CC2)cc(NS(=O)(=O)CCC(F)F)nn1 CCCC(C(=O)N(CC1CC1)CC)NC(N)=O.c1(C=O)cc(C(C)(C)C)ccn1 Cc1ccc(C=CC(N2C(CNC(=O)C(C)NC=O)CC3CCCC23)=O)cc1C C#CC1CCN(C(=O)COC(C)(C)CNC(C2(N3CCCC3)CC2)=O)C1 C(CC(C)C(=O)N(CC)CC1CN(C(=O)CCC=CC(C)C)CCO1)=CC C1(CCC)(NC(c2cnc(Cl)[nH]2)=O)CCN(C(=O)CNC(c2ccoc2)=O)CC1 c1(CC(=O)NCC(CC)NC(C2CCNC2=O)=O)ccc2c(c1)CCCS2 C1(NC(C=C(CC)C)=O)CC(CNC(=O)CCCc2cccs2)C12CCC2 CCC(C)(C)CC(=O)N1CCC(C(=O)NCC2CC23CC3(F)F)(CF)C1 c1(CC(=O)NCC(CCNC(C2(CSC)CCC2)=O)O)cc[nH]c(=N)c1 N1(C(CSCCC#N)=O)CC2CCOC2(CNC(=O)Cc2cnsc2)C1 Cc1cc(C(N2CCC(C(C)(C)C)(CNC(=O)CC#N)C2)=O)c(F)c(Br)c1 CC1CCN(C(=O)CC2CCSC2)CCN1C(C1CC2(CCOCC2)C1)=O C12(CNC(C(C)=C(C)C)=O)CCCC1CCN2C(=O)CCc1cnccn1 c1(C(N2CCC(N(C(CC3CCN(C)C3)=O)C)C2)=O)ccc(N(C)C)cc1 c1(C(=O)NCCCN(C(C(CCSC)N(C)C)=O)C(C)C)c(F)cccc1F CS(=O)CCC(=O)N1CCN(C(=O)Cn2nnc(-c3ccccc3)n2)CC1 C1(CNC(C(C)O)=O)(NC(c2cccc(C3OCCO3)c2)=O)CCOCC1 CC(C)CS(=O)(=O)CC(=O)N1CC(n2cc(CNC(=O)C(C)(C)F)nn2)C1 N1(C(C(c2cccc(Cl)c2)C)=O)CCC2(CC1)CN(C(C1(CF)CCC1)=O)C2 C#CCC(C(=O)NCC(N1CCCCC1)C)NC(=O)CN1CCSCC1 c1(C(N(C)CCOCCNC(=O)CC(C)(C)C#N)=O)cc2occ(Br)c2[nH]1 c1(N(S(=O)(=O)Cc2ccc(Cl)cc2)C)cnnc(O)c1Cl.C1CC2CNC1C2 c1(C(c2nnnn2CC)Nc2cccc(C)c2C)cc(OCC)ccc1.CCO Cc1cc(=NC(=O)C(=O)N(C)CC2CN(C(=O)C#CC3CCCC3)CCO2)[nH]o1 C1(C(=O)N(C2CCSC2)C)(CC)CCCN(C(=O)CCC(C)(C)N(C)C)C1 C1(CCNC(C2(OC)CCOCC2)=O)C(C)CCCN1C(=O)CCc1cnc[nH]1 C(=O)(CCCCC(F)(F)F)NC1CC2CN(C(c3cccc(OC)c3O)=O)C1C2 N1(C(CCNC(CC(C)C)=O)=O)CC(NC(C2CCCN2C=O)=O)CC(F)C1 c1(C(=O)NCCC(=O)Nc2ccc(OC)nc2)n[nH]c2c1CCC2C N1(C(c2cn(CCC)nc2C)=O)CC(CNC(=O)CC2CCOC2)C(F)(F)C1 N1(CC(=O)NCCC2CCC(CNC(CN(CCC)C)=O)C2)CCC(C)(C)C1 C(C)(C(CC(=O)NCCSCCCO)NC(c1cncc(F)c1C)=O)OC C(C1=CCN(C(=O)CCC2CCOC2)CC1)NC(c1ccccc1NC1CC1)=O C#Cc1cc(C(N2CCCC(N(C)C(C3CCC3(F)F)=O)CC2)=O)cc(F)c1 c12ccc(cc1)OCC(=O)NC(C)(C)CNC2=O.c1(N(S(C)(=O)=O)C)nncs1 C(=O)(CCC(C(=O)NCC(C)C)N1CC=CC(C(=O)OC)C1)OC S(=O)(=O)(c1ccc(C(=O)NCC2CN(C(c3nccn3C)=O)C3CC23)cc1)NC c1(C(N2CC3C(CNC(CCC=CC(C)C)=O)(C3)C2)=O)csc2cncn12 C1(C(=O)Nc2c(C(=O)OC)cc(Cl)c(OC)c2)CCC(F)(F)CC1(C)C N1(C(c2cc(C)on2)=O)CC(NC(c2ccc(Br)nc2O)=O)C2CCCCC12 C(CC(=O)NC(c1cncnc1)C)(C(F)(F)F)NC(C1C(OC)(OC)CC1)=O N1(C(Cc2nc(C)[nH]n2)=O)CC(NC(c2ccco2)=O)CC12CCC2 c1(C(=O)NC(CNC(C(CC(C)C)F)=O)C(C)C(C)C)ccc2cc[nH]c2n1 c1(OC)cnnc(C(N2CC(C(O)C(=O)N(C)Cc3cc(=O)cc[nH]3)C2)=O)c1 n1(CC(=O)N(C)CCN(C)C(C2(C)CC2(F)F)=O)nc2n(c1=O)CCCCC2 C(=O)(C(Cc1ccccc1)C(C)C)NCC1(F)CC(NC(CC=CC=C)=O)C1 C(=O)(C1=CS(=O)CCC1)NCCCN(C(=O)CCCc1cnccn1)CC Cc1cc(C(=O)NCC2CCC(C)CN2C(=O)Cc2cnsc2)cnc1C(F)F C(=O)(CC1OCc2ccccc21)NC(C)C(C)(C)NC(=O)Cn1ncn(C)c1=O Cc1ncc(C=CC(=O)NCC(C)CNC(=O)CSc2ccccn2)c(O)n1 c1(OC)cc(O)ncc1C(N1CC(NC(C2C3C4CCC(C4)C23)=O)C1)=O N1(C(C(C(=C)Cl)(C)C)=O)CC2CC(C1)CN(C(=O)CCSCC(N)=O)C2 C1(NC(C2(COC)CN(C(=O)CC3COCC(C)O3)C2)=O)CC2CCC1(CO)C2 C#Cc1ccc(N=c2scc(-c3ccco3)n2Cc2nn(C)cc2S(C)(=O)=O)cc1 C1(NC(CN(CC)CC)=O)CCC(O)CN(C(c2cnn(CC(C)C)c2)=O)C1 c1(C(=O)NCC2CCN2C(C2CC(N3CCCC3)C2)=O)cnoc1-c1ccco1 C1(CCNC(CC(C)OC)=O)CCCN(c2ncnc(=N)[nH]2)CC1 c1(NC(C)=O)ccc2c(c1)CN(C(=O)N=c1ccc(C(C)(C)C)n[nH]1)CC2 c1(CC(C)C)cc(C(N2CC(CNC(c3nccs3)=O)CC2C)=O)cc(O)n1 c1(OC)cccc2c(C(=O)NC(C)(C)CCNC(=O)C(C)C(F)(F)F)csc12 c1(OC)cc(C)c(C(N2CCNC(c3cc[nH]n3)C2)=O)cc1OC Cc1cc2sc(NC(=O)Nc3cccc(F)c3OC(F)F)nc2s1 Cc1cccc2[nH]cc(CCC(=O)NCC(O)CNC(c3cnc(S)n3C)=O)c12 Cc1cc(Br)ccc1-n1nc(CCC(C)C)nc1Cn1nccn1 C(CCC(=O)N(C1(CO)CCC1)C)N(C)C.C1=CCONC1=O CCCCC(C)(F)C(=O)NCCCCC(C)NC(c1ncc(Cl)cc1F)=O C#Cc1cc(C(N2CC(C(=O)NC(c3ncc(C)s3)C)CCC2C)=O)ccc1C N1(C(C(C)OCC#C)=O)CCCC1CC(=O)N(CCC(N)=O)C C1(C(=O)NC(C(=O)NC(C=C)(C)C)C)Cc2nccn2C1 CC(C)CC(C(=O)N1CC2CCCC(C1)N2C(C1(C#N)CC2CC2C1)=O)C(N)=O C1(NC(C(Br)=C(C)C)=O)CC(C)N(C(c2coc(-c3ccccc3)n2)=O)C1 CC1CS(=O)(=O)CCCN1C(C(=O)NCc1nnn(C)n1)c1cnsc1 CCCC(C(=O)NC1C2COCC12)NC(c1n[nH]c(C)c1O)=O C(=O)(CCCCCCn1cc(CNC2(C#N)CC3CCC2C3)nn1)OC C1(CC(=O)NC(c2cccc(C)c2)CNC(C(C)SCC)=O)CCCCCCC1 c1(C(=O)NC(C(=O)NC2(C#C)CCOC2)CC2CCCC2)ccc2cncn2c1 c1(C(=O)NCCCN(C(C(CC=C)C)=O)C2CC2)c(O)cncc1F c1(OCC)ccc(C(=O)NCCC(C)CCNC(=O)CCC2CCCN2C)cn1 N1(C(CCC)=O)CCC(C2CN(C(c3ccc(OC4CCCCC4)cc3)=O)C2)C1 N=c1ccc(C(=O)NCC2CC2NC(=O)COCc2cccc(Cl)c2)n[nH]1 C1(CNC(CCCC=C)=O)CC(C(C)(C)C)CN(C(=O)C(C)CC(N)=O)C1 CCCC(C(=O)NCCCN(C(=O)CC1CC1)C)C(C)C C1(CNC(c2ncccc2C(F)(F)F)=O)C2CCC(C2)N1C(=O)Cn1nccn1 CC1(C)CCC(Nc2cc(NCCc3cccc(Br)c3)ncn2)CN1 N1(C(CCC(=O)OCC)=O)CCOC(C)(CNC(C2(C(C)(C)OC)CC2)=O)C1 C1(NC(C(N2CC(F)CC(NC(=O)OC(C)(C)C)C2)=O)=O)CCCC12OCCO2 c1(CNC(=NC)NCC2CC(=O)N(C)C2)cc(Cl)c(Cl)c(Cl)c1 N1(C(CC2OCCN(C(c3c(C)c(Br)cnc3)=O)C2)=O)CCc2ccsc2C1 c12ccccc1N2.C(C)(C(=O)NC(CNC(=O)CC#N)CC)OCCC=C C12(c3cn(CCOC)nn3)CC(CN1C(c1cnc(-c3ccco3)s1)=O)C2 N1(C(c2cn(CC)nn2)=O)CC(C)OC2(CCN(C(=O)C(CO)N(C)C)CC2)C1 c1(CNc2c(OC)ncnc2)cccc2nn(C)cc12 N(C1CCCn2ccnc21)C(CC1CN(C(Cc2cc(C)n(C)n2)=O)C(C)C1)=O C1(CC(C)NC(c2cc(O)n(C)n2)=O)CCN(C(C2C(C)(C)C2(C)C)=O)CC1 CSC1=C(C(=O)N2CCC(NC(c3cnn4ccsc34)=O)C2)CCCC1 c1(C(=O)NCC2(C)CC(NC(=O)Cn3cnnc3)C2)ccc(F)cn1 c1(C(=O)NC2C=CC(C(=O)NCCCOC)C2)c(C(F)(F)F)ccc(Cl)c1Cl C1(C#N)(C(N(CC(C)NC(C2CCCS(=O)(=O)C2)=O)C)=O)CCOCC1 C(=O)(CCCS(C)(=O)=O)N1CCC(C)C1CNC(c1cc(=O)n(C)o1)=O C(C(=O)NC1CCC1CNC(c1ccc(C)c(C(C)(C)C)c1)=O)(C(C)(C)C)OC C1(CNC(C2CCCC2C(F)F)=O)CC(F)(F)CN1C(=O)Cc1ccnc(F)c1 N(C1CCc2ccccc21)C(C1CC(C)N1C(c1ccc(Br)cc1)=O)=O CCCC(O)(CCC)CC(=O)NCCCN(C)C(c1ccc(OC(C)C)cc1)=O N1(C(c2ccc(C#C)o2)=O)C2CCC1C1CC1(NC(=O)CC1CCCC13CC3)C2 c1(CC)cc(C(=O)NC2(CN(C(=O)C(C)OC)C)CC2)cc(Cl)c1 S(=O)(=O)(CCN=c1[nH]c2c(c(=NC3CC(C(F)(F)F)C3)[nH]1)CSC2)NCC c1(CNC(=NCc2cc(C)on2)NC2CC2C)csc2ccc(Br)cc12 c1(NC(C2CCCN(c3ncc(C4CC4)cn3)CC2)=O)n[nH]c2c(F)cccc12 Cc1ncc(N)cc1C(=O)NC(CNC(C1CCCS(=O)(=O)C1)=O)C(C)(C)C Cc1c(C(N2CCC2c2ccncc2)=O)nnn1CC1COCCO1 C1(CNC(C2(CC)COC2)=O)CC2(CC2)CN1C(=O)Cn1cnnn1 C1(C(CN(C2CCCC2)C(N2CCC(N(C)C)C2)=O)N)CCC(F)(F)CC1.CCS N1(C(c2c(C#N)nc(C)o2)=O)Cc2[nH]nc(-c3cncnc3C)c2C1 CC1CN(C(=O)CCOCCCN(C)C)CC1CN=c1[nH]ncs1 Cc1ccc(C(N2CCCC(O)(CNC(c3ccncn3)=O)C2)=O)c2c1CCC2 CCCC(CC)C(=O)NCCCC1CN(C(C2(C#N)CCC2)=O)CCO1 Cc1cccc(C(=O)NCC2CC(C)N(C(C3(C)CCCCCC3)=O)C2)c1O C12(NC(C)=O)CCCCCC1N(C(c1cc3sc(C)cc3s1)=O)CC2 CC(C)CC(CO)CN=c1ccc(S(=O)(=O)NC(C(C)(C)C)C2CC2)c[nH]1 C(CCCCOC(c1cn(CCNS(N)(=O)=O)nn1)=O)NC(C)(C)C O=S(=O)(c1cc(Cl)ccc1Cl)N1CC(NCc2ccc(Cl)cc2Br)C2(CC2)C1 Cc1ccccc1C1=NOC(C(N2CC3C(NC(=O)C=C(Cl)Cl)C3C2)=O)C1 C=CC1(C(=O)NCCC2CN(C(C3CCCS3)=O)CCO2)CCCCC1 Cc1c(NC(=O)CC(O)CNC(=O)CC2CCOC2(C)C)cccc1C#N N1(C(Cc2cc(COC)on2)=O)CCCC1(C)CNC(C1CCSCC1)=O c1(C(=O)NC2CCN(C(CC(CC)OC)=O)CC2O)c(C)nn2cccnc12 C(c1ccc(F)c(F)c1)=C(C)C(N1CC2CC1C2NC(c1cnc(O)s1)=O)=O C1(C(N2CCC(CC)C2CNC(C2CCOC2(C)C)=O)=O)CCCCCCC1 C(=O)(C(C)(C)C(=O)NC1CCN(C(=O)CC2CCCSC2)CC1OC)NC C1(NC(CNS(NC)(=O)=O)=O)CCN(C(c2sc(NC3CC3)nc2C)=O)CC1O c1(NCC)ccc(C)cc1C(=O)NC1CCN(C(c2ccccc2F)=O)C1 C1(C(N(C)CC2CCN(C)C2)=O)CCCCCCN1C(=O)CC1(O)CCOC1 C1(NC(COCCC)=O)CCN(C(c2ccn(C(C)C)n2)=O)CC1C Cc1n[nH]c(C)c1C(=O)NC(CO)C(C)NC(C1CC(F)C1)=O N1(C(c2c(CC)scc2)=O)CC2OCC(NC(=O)CN3CCC(C)C3)C2C1 c1(C(C)=O)cccc(OCC(N2CCCC(NC(c3cc(Cl)cs3)=O)C2)=O)c1 C1(CC=C)(NC(=O)COCc2ncnn2C)CCN(C(=O)C(F)C(C)C)C1 C1(CCC(=O)N(C(C)(C(=O)NC2(CCCF)CC2)C2CC2)C)NC(=O)NC1=O N1(C(c2ccncc2N2CCOCC2)=O)CCCC(O)(c2ccccc2)CC1 C1(CC(=O)NC(CNC(c2cnc(CC)[nH]2)=O)CC)CCCC(F)(F)C1 N1(C(C(C)CF)=O)CC(CNC(=O)COc2cccc(Br)c2)CC(C)(C)C1 c1(C(C(=O)NC(CC)C)N(C)CC2CC3CCC2CC3)ccc(OC)c(OC)c1 c1(C(=O)NC2CC(F)(CNC(c3cnc4n3CCC4)=O)C2)cccc2c[nH]nc12 C1(C)(NC(C(CO)OC)=O)CCCN(C(c2cncc(F)c2)=O)C1 S(=O)(=O)(c1cccnc1)N1CC(NC(C2(C(C)C)CCC2)=O)C2(C1)CC2 C1(NC(c2ccc(C(N)=O)s2)=O)CCCN(C(=O)C2=C(Cl)CCC2)CC1 c1(C(N(C)CC2CCCN2C(=O)CC2CCOC2=O)=O)cc2ccncc2[nH]1 c1(NC)ccc(C(=O)NC23CC2CN(C(=O)Cc2cccc(C4CC4)c2)C3)nc1 N1(C(c2c(C(C)C)noc2)=O)CCc2sc(CNC(=O)CCC#N)nc2C1 n1(C2CCCN(C(CC(CN)O)=O)C2)cnc2cc(Br)ccc12 N1(C(=O)Nc2cccc(CS(=O)(=O)c3ccccc3)c2)Cc2cccc(CO)c2C1 Nc1cccc(C(=O)NCCCNC(C2CC(F)(CF)C2)=O)c1F N1(C(C(CC)OCC)=O)CCC(C=CC(N2CC(CO)C(C)(C)C2)=O)CC1 C(C(O)CC(=O)NCC(C)(C)C1CC1)NC(c1nc(CCC)oc1)=O n1(CC(N2CC(C3(NC(C(C)OCC(C)C)=O)CC3)C2)=O)nnc2ccccc12 C(=O)(CCC(=O)NC(C)C(c1ccccc1)NC(C1CC(N(C)C)C1)=O)NC c1(OC)cc(Br)c(Cl)cc1C(=O)NCC1CC1c1ccc(C)nc1Cl N1(C(C23C(=O)C4CC2C3C4)=O)CCOC(COCC)CC1.C123CC(C1)(C2)NC3=O C1(C(=O)NC(C2(C)CCN(C(=O)CCN(C)C)C2)C)C2CN(CC(F)(F)F)CC12 C1(CC(=O)NC2CC(C)(NC(C3C(C)(C)CC3)=O)C2)Cc2ccccc2NC1=O CN1C(=O)CC(c2nc(-c3cccc(Cl)c3)nn2Cc2ccsc2)NC1=O n1(CC)ccc(C(=O)NC(C2CCCN2C(=O)CCc2ccsc2)(C)C)cc1=O N1(C(Cn2ccc(C)n2)=O)C(C(=O)NOCC2CCCO2)C2CCCC12 C1(CCNC(C=C(CNC(c2cc(CC)[nH]n2)=O)C)=O)NC(=O)NC1=O C1(NC(c2cccc(O)n2)=O)CCC2(CC1)CCN(C(c1cccnc1O)=O)C2 C1(NC(C2N(C(C3C(C(C)(C)C)CC3)=O)CCC2)=O)CCCC2(C1)N=N2 c1(C(=O)NCCN(C(C2CC2OC(C)=O)=O)CC)sc(C)nc1C C1(CNC(CCCCC)=O)CCC2CN(C(c3nn(C)cc3C)=O)CC12 c1(C(N(CCCNC(c2cc(C)n(C3CC3)n2)=O)CC)=O)cc(C)cc(C)c1O Cc1cc(C(=O)N(C2CCN(C(=O)CC3CC3)C2)C)n2ncnc2n1 C1(N(C(=O)NCC2(CO)CC23CCC3)CC)Cc2cscc2C1 C1(CC)COCCN(C(=O)Cc2ccc(C(C)C(F)(F)F)cc2)C1 C(=O)(C(C)CCNC(=O)C(=O)Nc1ccc(Cl)nc1)OC c1(CC)ncc(C(N2CC(C(O)C(=O)N(C)CC)C2)=O)o1 c1(C(N2C(C)CCC2C(=O)NC(C#N)C(N)=O)=O)cccc2cc(Br)cnc12 C1(O)(C(=O)NCC2(F)CC(NC(C(C(C)C)OCC)=O)C2)CCC(C)(C)CC1 c1(NS(=O)(=O)Cc2cccc(F)c2)ccc2c(c1)CCCC2O c1(CNC(C(C)SC)=O)cnn2c1CN(c1nnc(SC)s1)CC2 N1(C(CNC(=O)OCC=C)=O)CCC2C(C1)CN2C(=O)CC(C)n1ccnc1 C(=O)(CCCCCCS(N)(=O)=O)NC(C(C)NC(C(C)SCC)=O)C c1(CN(C(C(C2CC(NC(C(C)=C3CCC3)=O)C2)F)=O)C2CC2)ccccc1 N1(C(C2(OC)CCC2)=O)CCCC(C(C)C(=O)NOCC(F)F)C1 C(CCCC(=O)NCCN(CCOCCO)C(C1CCCS1)=O)N(C(C)=O)C N1(C(C2C(C=C)CC2)=O)CCC(NC(c2sccc2C(F)F)=O)C(O)C1 C(=O)(CCCCCO)N1CCCC(C(C)NC(CCc2ccc(C)cc2)=O)C1 N1(C(CCCNC(C(C(C)C)F)=O)=O)CCN2CC(F)CC2C1 C1(C(=O)NCC(C)(C(C)C)NC(C(CCC)NC(C)=O)=O)CCC2(CCC2)CC1 c1(CNCC(COCC(C)C)O)ccc(C(C)(C)C(=O)O)cc1 C(=O)(C(F)CC(C)(C)C)NC1(COC)CCCN(C(c2ccsc2C#N)=O)C1 c1(NCC2N(C)CC(O)CC2)c(F)cc([N+](=O)[O-])cc1F C(CC(C)(C)C(=O)NC(CNC(c1cc(F)cnc1OC)=O)C(C)(C)C)OC C1(C(N(CCN(C(=O)Cc2ccccc2F)C(C)C)C)=O)OC2CCC1C2 c1(C(=O)NC(Cc2cn(Cc3onc(C(C)OCC)n3)nn2)C)cnnc(O)c1 N1(C(C(C=C)c2ccccc2)=O)CCN(C(=O)Cc2cnn(C)c2C)CC1CC O=C(C1CCCCc2ccccc21)NC1C2CCN(C(=O)C=C3CCC3)C12 CC1(C(N2CC(CNC(c3cc(Cl)c(Br)[nH]3)=O)C(O)C2)=O)CCC(=O)N1 c1(C(=O)OC)cc(F)cc2c1CN(C(C1CC3(C1)CC(C)(C)C3)=O)CC2 C(=O)(C1=NOC(CNC(C2CCC(=O)C2)=O)C1)N(CC(=O)NC1CC1)C C(CCO)(C(=O)NC1CCCN(C(=O)C(C)(C)n2cc(Cl)cn2)C1)N(C)C C1(C(N(C(C)CNC(=O)C(C)(C)N2CCCC2)C)=O)CC(=O)N(C)C1 CC(O)C(C(=O)N1CCN(C(c2cc(-c3ccc(F)cc3)no2)=O)CC1)N(C)C N1(C(C2(C3N(C(CC=CCC)=O)CCC3)CC2)=O)CC(=O)N(C)CC1C N1(C(C2C(C#N)C2)=O)CCC2(CC1)COCC(CNC(c1c[nH]cc1Br)=O)O2 c1(SC)ccc(O)c(C(=O)NCC2CCCCN2C(C2CCCCS2(=O)=O)=O)c1 C=CC1(C(=O)NC(C)Cc2cnn(C)c2)CCN(C(C2CCCCS2)=O)CC1 C(C1c2ccccc2CCN1C(=O)CC1CCCCC1)NC(COCCSC)=O O=C(C#CC1CCCCC1)NC1CN(C(C2CC3CCC(C2)O3)=O)C1 CCCCS(=O)(=O)CC(=O)N1CCOC2CN(C(c3ccsc3C#N)=O)CC12 c1(-c2cn(CC(N3CC(SCC)C(N(C)C)C3)=O)nn2)ccc(Cl)c(OC)c1 C1(N(C(C2(CCC)CCC2)=O)C)CCN(C(=O)CCC2CCC(C)O2)CC1 Cc1nn[nH]c1C(N1CCC(N(C)C(c2cnn(C3CC3(F)F)c2)=O)C1)=O CC1CCN(C(c2cnc(-c3ccco3)s2)=O)C1CNC(=O)CCC(C)O CC(C(=O)NCC(C(C)(C)C)NC(c1ccncn1)=O)C(C)(C)O CC1CN(C(C=Cc2ccccc2)C(=O)NCC(F)F)CCS1 C1(C(=O)NCCCP(C)(C)=O)C2CCCCCCC12 c1(-c2nc(CC(C)OC)nn2-c2cnnn2C)ccc(OC)c(C(C)C)c1 N1(C(CCOC(C)C)=O)CC(NC(c2ccn(C(C)C)n2)=O)CC12CCCCC2 c1(C(N2CCN(C(CN(C3CC3)CC)=O)C(CO)C2)=O)ccnc2[nH]nnc12.C1CC1 c1(C(=O)NCC2(N(C)C)CCC2)cc2c(-c3ccn4cnnc4c3)cccc2[nH]1 c1(C(N2C(C)CC(NC(=O)Cn3ccnn3)CC2)=O)noc2ccccc12 c1(CC)nc(C)c(CC(=O)NC2CS(=O)(=O)CC2NC(=O)C=CCF)c(C)n1 C(=O)(CC(CC)C(F)F)NCCC1(O)CN(C(C2CC(OCC)C2)=O)C1 N1(C(CC2CCN(C(C(COC)N(C)C)=O)CC2)=O)CCC(O)C(C)C1 c1(C(=O)OC)nn(C)nc1C(=O)NC1CCN(C(=O)CCCN(C)C(C)=O)CC1 C=CCCC(F)(F)C(=O)N1CCC(N(C(=O)C=Cc2cnn(C)c2)CC)C1 N1(C(CCCC)=O)CC(CNC(C2CCN(C3CCCCC3)C2)=O)C(C)(C)C1 c1(C(=O)NCC2CN(C(CCCC(C)=O)=O)C(C)C2)cc2ccccc2oc1=O O=C(C(Cl)=CCl)NC(CNC(=O)Cc1cc(C2CCC2)no1)C1CC1 Cn1ncc2c(C(N3CC(CNC(C4CC(=O)NC(=O)N4)=O)C3)=O)ncnc12 c1(CC(=O)NCC2(CN(C(C3(COC)CCC3)=O)C)CC2)csc(Cl)n1 C1(C(N2Cc3c[nH]nc3C2)=O)CC2CCC(C1)N2C(=O)C(F)(F)C(F)F C#CCC(CC#C)C(=O)N(CC(C)(C)CNC(=O)C(C)CN(C)C)C CC1(F)CN(C(c2cc(C(F)(F)F)n[nH]2)=O)CCN(C(C2(O)CCSC2)=O)C1 C(=O)(C1c2c[nH]nc2CN1C(c1cc(C#N)cn1C)=O)N1CCC(OC)C1 C1(=C(C(=O)NCC(CNC(C(C)=CC)=O)C)F)CCCCC1 c1(C(N(CCCN(C)C(C2CC2c2nc[nH]n2)=O)C)=O)ncoc1C1CCCO1 C#CC1COCCN1C(C1(N(C(=O)C=C(C)COC(C)=O)C)CC1)=O N1(CCCC)CCOCC1C(N1CCC(C(C)NC(=O)OC(C)(C)C)CC1)=O c1(OC)cccc(OC)c1CC(N1CC2CC1(CNC(=O)CC1CC1C)C2)=O C(=O)(C(F)C(C)(C)O)N1CCC(C(C)NC(=O)CN2CCOCC2=O)C1 N1(C(Cc2ccc(C(=O)OC)o2)=O)CCOC(CNC(c2[nH]ccc2C)=O)C1 C(CN=c1[nH]nc(C#N)s1)Nc1nccc(=NCC2CC(C)SCC2)[nH]1 C1(CNC(CC)=O)CC(OC(C)C(=O)NC)CN1C(c1nc(OC)c(C)s1)=O N1(C(=O)NC(C)C)CCCCC(NC(N2CCOC(C(F)F)C2)=O)C1 c1(NC(N(C(CCCC)C)C)=O)c[nH]cc(C)c1=O c1(C(C(=O)NC(C)(C)C)N(C(C(=O)OC)C)C(C)(C)C)sc(NC(C)=O)nc1C N1(C(c2ccc(COC)[nH]2)=O)CC(CNC(C2CCC2)=O)C(O)C1 N1(C(C)C(=O)N(C)C(c2nccs2)C)CCN(CCCC#N)CC1 C1(C)(CC)CC(NC(c2cccnc2)=O)CN1C(=O)Cc1cccc(F)c1OC C(=O)(CCCCCCBr)N1CCC(CNC(=O)Cc2ccnc(Br)c2)C1 C(=O)(C(F)C(C)CNC(=O)C(C)n1ccnn1)NC1(CCCC)CC1 c1(C(=O)NC(CC(C)NC(C2CCC(C)CC2)=O)C)cnc2sccc2c1 N1(C(c2c(Cl)cnc(OC)c2Cl)=O)CCOC2CN(C(=O)CCC(N)=O)CC12 c1(C(=O)NC(C2CCN(C(c3cccnc3O)=O)C2)C)c(Cl)ccnc1F c1(C(C(=O)NCC(C)N(C(c2ccc(C)cc2)=O)C)(C)C)ccc(F)c(F)c1F N1(CCC(N)=O)CC(=O)N(CCCCO)C1 N(C1CCCc2ccccc21)C(COCC(NNC(c1c[nH]c2ncc(Br)cc12)=O)=O)=O C1(OC)(CNC(=O)C(F)(F)C2(OC)CCCC2)CCN(C(=O)C(O)C(C)C)C1 N1(C(c2cn(C)nn2)=O)CCN(C(C2CCCCS2)=O)CC1c1ccccc1 C1(C)(CCC)CCN1C(=O)C(C)NC(=O)C(C)c1ccco1 CCC(CC(=O)NCC1(CO)CC1(C)C)NC(=O)Cn1cc(C)cn1 Cc1snnc1C(=O)NC(C)C(C)(C)NC(=O)C(Cc1ccsc1)NC=O C(C(C(=O)NCC(CO)NC(=O)CNC=O)NC(C)=O)OC.C(C)(C)(C)O CC(C)CCC(F)C(=O)NCCC1COCCN1C(=O)C(O)CN(C)C N1(C(C(n2ncc(C)c2)C)=O)CCOCC(C)(CNC(=O)Cc2ccsn2)C1 C1(NC(=O)NC2CC(c3ccccc3)(NC(=O)OC)C2)CCC(C)N(Cl)C1 N1(C(C(C)(O)C(F)(F)F)=O)CCC2(CCC(NC(c3cnon3)=O)CC2)C1 Nc1cc(C(=O)NC2CCCN(C(c3occc3C3CC3)=O)CC2)cc(F)c1O C12(C(N3CC4C(NC(C(C(CC)CC)C)=O)C4C3)=O)CC3CC(C1)CC(C)(C3)C2 CC(C)CC(CNC(C1(F)CC=CCC1)=O)C(=O)NCCc1cnccn1 O=C(C1=CCCN(Cc2cc(Cl)ccc2Br)C1)NCCc1c(F)ccc(I)c1F C1(NCCC(=O)OC(C)C)CC=CC1O C1(C(=O)NC(c2cn(C)nn2)C(=O)NC2C(C)CN(C)C2)CC2(C1)CC21CC1 CC1CCC2(CC1)CCN2C(=O)C=CC1CCN(C(=O)CP(C)(C)=O)CC1 c1(C2(NC(C(C)N(C(=O)COC(=O)C=O)CC)=O)CC2)ccc(O)cc1 CC1CCN(C(c2conc2C2CC2)=O)CCN1C(c1ccn2cncc2c1)=O CC1(C)CC(C(=O)NCCC2(C(N3CC(CO)C3(C)C)=O)CC2)CCO1 c1(C(=O)NCC(N(C(CCC2CCCN(C)C2)=O)C)C2CC2)cccc(N)c1F Cc1cc(Cl)ncc1C(N1CCN(C(c2ccc(O)cc2Cl)=O)CC1)=O C(CCCCCNC(c1cc(COC)cn1C)=O)NC(C1C(C)(CC)C1)=O N1(C(COc2c(CC)cccc2)=O)CC2CC(NC(C3CC(C)(C)C3)=O)CC1C2 C1(C(N(C2CC(C#N)C2)CC(=O)NCC(COC(C)C)O)=O)CCC(=O)N(C)C1 c1(OC)cc(NC(C2(C)CCN2C(C2(F)CCC2)=O)=O)cc(OC)n1 Cc1cnc(C(c2nnnn2CC2CC2)NCC2(CO)CCCC2)c(C)n1 CCCC(C(O)C(=O)NC(CO)CCF)NC(=O)CCCNC(=O)NC C(CC(C)C)(C(=O)NC1CC(O)(CO)C1)NC(CC1CC(=C)C1)=O Cn1ccc(C(N2CCN(C3CCCN(C(C4CC(O)C4)=O)C3)CC2)=O)cc1=O C1(NC(CC(=C)C)=O)CC2CCCC(C1)N2C(=O)CC(O)CC CC1CCN(C(=O)CCn2ccccc2=O)CC1NC(=O)CC1CCSCC1 N1(C(C2CN(C(C3CC4CC4C3)=O)CC2F)=O)CCC(F)CC1 c1(C(=O)NC(CNC(c2cc(C)c(Cl)cc2F)=O)(C)C)csc2c(O)ccnc12 Cc1cc(N(C2CC23CCC3)CC2CN(C)CCN2C(=O)OC(C)(C)C)nc(Cl)c1 C1(C(N(CCC(=O)NCC(C)(C)SC)CC)=O)CC2CC(=O)C1O2 N1(C(CC(C)C(C)(C)C)=O)CC2(CCN(C(=O)C=Cc3ccccc3)CC2)C1 C1(C(N(CC(C)(C)O)C)=O)CCOCCN1C(=O)CCN=[N+]=[N-] C(=O)(C1=CCOCC1)NC(CCSC)C(=O)N1CC(c2nn[nH]n2)C1 Cc1ncccc1CC(N1CCC(CF)(NC(=O)CCCN(C)C)C1)=O C1(C(N(CCNC(c2cncc(OC(F)(F)F)c2)=O)CC)=O)CC(F)C(=O)N1C N1(C(CCCc2onc(C)n2)=O)CC2(CC(NC(=O)CCSC3CCCC3)C2)C1 C=CC1CN(C(C2OCCC2CC)=O)CC1NC(c1ccnn1CCCC)=O c1(CNC(C(c2ccco2)N(C)C(c2nc(=N)cc[nH]2)=O)=O)nn(C)c(=O)n1C c1(CC(=O)NCC(C)N(C(C(=O)NCC)=O)CC)cccnc1F Cc1ccc(NC(=O)COC2CCN(C(=O)CCC(N)=O)C2)cc1F Cn1nc(C2CC2)cc1C(=O)NCC1COCC1NC(c1ccc(Cl)cn1)=O N1(C(C(=O)NCC=C)CC2CCCCO2)CCC(O)(c2cnnn2C)CC1 c1(C(=O)NC(c2ccc(OC)cc2)C(=O)O)ccc(S(C)(=O)=O)cc1NC c1(C(=O)NCC2C(C(=O)Nc3c(C)scc3)CCC2)cc(O)cc(F)c1 c1(NCC(C)NC(C2C(OC)CCCC2)=O)ncc2c(n1)CCOC2 c1(C(N2CC(C(C)NC(=O)CCN3CCCC3=O)C2)=O)cncc(F)n1 C(C(C)NC(=O)C(=O)N(CCCN(C)C1CC1)C)(OC)OC N1(CC(=O)NCC(CCOC)NC(c2ccccn2)=O)Cc2ccccc2C1 CC(C1CC1)=CC(=O)N(C)CCOCCCN(C(=O)C(O)C1CC1)C Cn1nc([N+](=O)[O-])c(Cl)c1C(=O)NCC1CC(NC(=O)C(O)CC2CC2)C1 CC1CCSCCN1C(C1CC(C)(NC(C2CNC(=O)O2)=O)C1)=O C(=O)(C(C)(C)CCF)NC(CCC)C1CC1 N1(C(C2C(C)(CC)C2)=O)CC2(C1)SCCC2NC(=O)C=Cc1ncc[nH]1 n1(C(C)C(=O)NCCC2(NC(=O)C#CC(C)(C)C)CC2)c(=O)oc2ccccc12 c1(CC(=O)NC2C(NC(C(F)OC)=O)C2)ccccc1C C(=O)(CC(C)(C)n1cc(CCN2CCCC2)nn1)NC(c1c(CC)n[nH]c1)C N1(C(c2nn(C)cc2Br)C(=O)NCC(=C)C)CC(COC)OC(CC)C1 N1(C(C2=C(C)OCCS2(=O)=O)=O)CCCC2(CCCN2C(=O)Cn2cnnc2)C1 N1(C(CCC(C)SC)=O)CCN(C(=O)CS(=O)(=O)CC2CCCO2)C(CO)C1 C(=O)(C1Cc2ccccc21)N1CC(O)(CN(C)C(C2CC(C#N)C2)=O)C1 Cc1cnc(C(N2CC3C(NC(c4cc(C(C)C)ccc4C)=O)C3C2)=O)c(F)c1 C(=O)(CCC(=O)N1CCCC1C(C)(C)NC(C1(C)CCOC1)=O)c1ccc(C)s1 c1(OC)ccc(CNC(C2CN(C(=O)Cc3ccsc3)CCO2)=O)c(Cl)c1OC c1(NCc2cccc(C(=O)OCCC)c2)ccc(-c2ccccc2SC)cc1F C1(CC(=O)NC2C3CC(NC(C4(O)CCCCCC4)=O)CC23)CCCC2(CC2)C1 c1(C(N2CC(NC(C(CC)C#N)=O)C(OC)C2)=O)cn(C)c(=O)n1C C(=O)(C1=NNC(=O)CC1)NC1CC(CCNC(c2c(C)n(C3CC3)nc2)=O)C1 N1(C(CC(CCC)C)=O)CCN(C(=O)C=Cc2ccc(=O)n(C)c2)CC(O)C1 S(=O)(=O)(c1ccc(C#N)c(NCC2CC2(F)F)c1)NCC1(C(C)C)CC1 N1(C(CCC(C)(C)C)=O)CC2OCCN(C(=O)CC3(C(F)(F)F)CC3)C2C1 C(N=c1nc(N2CCC2)c2[nH]ccc2[nH]1)C1C(C)(C)CCCC1.C12CC3(CCC3)C1N2 Cc1ccc(F)c(C(=O)NC2CN(Cc3c(Br)ccc(C)c3F)CC2C#N)c1Br N1(C(C2C(NC(=O)Cc3nc(O)n[nH]3)CC2)=O)CCN(C(=O)C2CC2)CC1 C1(C(=O)NC(C(=O)NC(C)Cc2cn[nH]c2)CC2CCC2)C2CCCOC12 C(N=c1[nH]c(=NCCN2CCOCC2CC)[nH]c2c1CSC2)C1(CCC)CCC1 C=C(C)CCCC(=O)N(CCNC(c1cc(-c2ccc(Cl)cc2)on1)=O)CC N1(C(c2cc(O)nc(O)n2)=O)CC2(C(N3CCCC4(C3)N=N4)=O)CC1CCO2 N1(C(CSc2ccc(C)cc2)=O)CC2CC(C)N(C(C3SCCS3)=O)C2C1 C1(C(=O)OC)C(F)(F)C12CC(C(=O)NC1CC(NC(=O)C#CC(C)C)C1)C2 N1(C(C(C)C2CCC2)=O)CC(N(C(=O)CSC2CC2)C)C(O)C1 N1(C(CC(CC#C)NC(=O)CC2CC3CC3C2)=O)CCC(C)CC(C)C1 N1(C(c2cc(C#C)cc(N)c2)=O)CCC2(COC(CNC(c3cncs3)=O)C2)C1 CC(F)(F)C(C)(C)C(=O)N1CCCC(O)(CNC(=O)C(O)CC(F)F)CC1 CC(C)CC(CC(=O)N1CC(NC(c2sc3ccccc3c2Cl)=O)C1)CC(N)=O C1(CNC(C2N(C(C)=O)CCC2)=O)CC(C)N(C(=O)C=CC(N)=O)C1 Cc1c[nH]cc(C(=O)NC2CC2CNC(=O)CCCOC(=O)C(C)C)c1=O Cc1nnc2n1CC(C(N1CCC3CN(C(=O)COC(F)F)CCC13)=O)N(C)C2 C1(NC(C(COC)O)=O)COC2(C1)CN(C(=O)C1=C(Cl)CCOC1)C2 Cc1noc2nc(C(=O)NCCOCCN(C)C(c3nncn3C)C)ccc12 Cc1ccc(C(C)C(N2CC(CNC(=O)C=CCF)C(O)C2)=O)cc1 c1(NC(=O)C(C)(C)CF)ccc(CNCCCN(C(CSCC(C)C)=O)C)cc1 C(=O)(CCC(=O)C(C)(C)C)NC(CC)CCC(N1CCC(C2(C)CC2)C1)=O N1(C(CCC=C)=O)CCC2CC2(C(=O)NCC(C)(O)CO)CC1 C12(NC(CCc3ccc(C)s3)=O)CCCC1N(C(=O)C1=CCC(C)CC1)CCC2 C1(C(N(CC(CN(C)C)O)C)=O)CC2CC1CN(C(C1C3CC4C(C3=O)C14)=O)C2 C1(NC(c2cnc(COC)s2)=O)CN(C(c2cc(OC)cnn2)=O)CC2(CC2)C1 c1(C(=O)NC2CN(C(c3scc(C)c3Cl)=O)C(C)C2)cnc2occc2c1 C1(NC(Cc2c(C)n[nH]c2C)=O)CN(C(=O)CCC2CCC(=O)N2)C(C)(C)C1 C1(CC)CCC(C)N1C(C1CCCN(C(=O)C(OC)OC)C1)=O c1(C(=O)NCC2C(CNC(c3cc(C)sc3C)=O)C2)ccc2c(c1)CCO2 C1(C)(C(=O)NCCN(C2CC2)CC)CC(O)CN1C(=O)CCC1CC1C CCC(C)CC(C(=O)NC1(C(=O)OC(C)C)CC1)NC(=O)C=Cc1cnc(C)s1 C(N=c1[nH]c(=N)[nH]c(=NC2CCCSCC2)[nH]1)c1nc(CC)sc1 c1(-c2ccc(CNC(C(CC)n3ccnc3)=O)cc2)c2ccccc2nn1C C1(NC(c2cn(CCC)nc2)=O)CCN(C(c2ccc(F)cc2F)=O)C1(C)C N1(C(C(F)=CCC)=O)CCC(C2CC2)C1CNC(=O)C(C)(C)C1CCCCC1 C1(NC(C(C)CC2CCC2)=O)C2CC3CN(C(=O)CC4CC45CC5)C1C3C2 N1(C(C(C)(C)C)=O)CCOC(C(=O)NC2CC2CNC(c2csnn2)=O)C1 CCCCCCCCCC(=O)N(CC(CC)NC(C1(n2ccnn2)CC1)=O)C C1(NC(c2c(C(N)=O)coc2)=O)C2CN(C(c3ccc(O)nn3)=O)CC12 C12(CC(=O)Nc3c(C)nn(CCF)c3)CCC1CN(C(=O)Cc1ccc(F)cc1)C2 C(=O)(C1=CCCOCC1)N1CCC(C)C(CNC(C2CC=CC(O)C2)=O)C1 CC(C)CCCCCC(=O)N1CCCC12CCN(C(C1CCCC(=O)O1)=O)C2 c1(N2CC(C(C)C)OCC2)ccc(S(=O)(=O)NC2(C)CCCCC2(F)F)cn1 C1(CCNC(=NC)NCCC2(C3CC3)CCCO2)CC(C)(C)CO1 C(C)(C(=O)N(C1CCN(C(c2c(C3CC3)cnn2C)=O)C1)C)(C(C)C)NC(C)=O C1(C(F)F)(CNC(C=CCC)=O)CCN(C(C2CCCCN2C(=O)C(C)C)=O)C1 c1(C(=O)NCCNC(=O)OC(C)(C)C)cc(C2(C)CC2)ccc1F.N12CCC(C1)C2 C(=O)(C1=CCC(C)CC1)N1CCC(C(C)C(=O)NC(C)(C)CO)CC1 C=C(Cl)C(C)(C)C(=O)NC12CC1CN(C(C1CCCCN1C)=O)C2 C1(C(=O)NCC2C(C(=O)NC(C=C)C)CCCC2)CCC(C#N)CC1 c1(OC)ccc(Br)c(C(N2CCC(F)(C(N3CCOC(O)C3)=O)C2)=O)c1F c1(CN(C(c2ccc(OC)cc2)C(=O)OC)C)ncc(Br)c(OC)c1C c1(C(=O)NCc2cccc(NC(CCOCC(C)C)=O)c2)occ2c1CCOC2 CCC(C)CC(C(=O)NC1(C)CCC2(CC1)CC2)NC(=O)Cc1cccc(F)c1 C1(C(N(C2(c3cc[nH]n3)CC2)C)=O)CCOC1CNC(=O)CCOC1CCC1 C1(C(N2CCC(OC)C2)=O)CN(C(C2(CSC)CC2)=O)CC1F c1(OC)cnc(C(=O)NC2CCCC(CNC(=O)Cn3nnc(=N)[nH]3)C2)c(F)c1 c1(CC)cc(C(=O)NC2CCC(CNC(c3nccn3C(C)C)=O)C2)ns1 N(C)(C1=NS(=O)(=O)c2ccccc21)C(C#C)C(=O)N1CCC(OC)C1 N1(CCC(=O)NC(C2CCCC2)CNC(CC)=O)CCN(CC2CCN(C)C2)CC1 C1(CNC(Cn2c(=N)scc2)=O)CN(C(=O)Cn2cnnn2)CCO1 CC1CN(C(=O)CP(C)(C)=O)CC1(C)CNC(c1ccc(C(C)(C)C)o1)=O CC(C)(C#N)CC(=O)N1CCCC1C1(C(=O)NCC2=CCCCC2)CC1 CC1CCCC(C(=O)NCCN2CCN(C(C3CC(n4cnnc4)C3)=O)CC2)O1 N1(C(CC2(COC)CCCC2)=O)CCN(C(=O)CS(C)(=O)=O)CC1c1cn[nH]c1 c1(C(N2CC(NC3CCOC3)C2)=O)coc2c(F)cc(F)cc12 C1(CNC(CCOC)=O)CC2CCC1N2C(=O)C(Cc1ccccc1)N(C)C CC1CN(C(C2(C(F)F)CCOCC2)=O)CCC1NC(C1CCC(C)C1)=O C(=O)(C(F)(F)C(F)(F)F)N1CCC(CNC(Cc2cccc(SC)c2)=O)C12CC2 N1(C(c2c(C)nsc2)=O)CC2(C1)CN(C(=O)C(C)OC1CCCCC1)C2 CC(C(=O)NC1CCCN(C(c2ccc(N(C)C)nc2)=O)CC1)C(C)(C)C C1(C(=O)NC)CCN(C(C2(C)CCN(C(C3CCC(OC)CC3)=O)C2)=O)C1C c1(NC(C(=O)NCCS(=O)(=O)N(C)C)=O)cccc(-c2cnn(C)c2)c1 N1(C(CCCCC#C)=O)CCCC2C1CCN2C(C1CC(C)(C(C)(C)C)C1)=O CC(C)C(CC1CCCCC1)C(=O)NCC(CO)NC(c1ccc(F)cc1N)=O C1(C(N2C(C)(CC)CC(NC(=O)COc3ccsn3)C2)=O)C2(CCC2)C12CCC2 c1(CCNC(=O)CC2CCN(C(=O)CCCn3ccnc3)C2)ccc(O)nc1 C1(NC(C2CC(=O)N(C3CC3)C2)=O)COCCN(C(c2ccc(Cl)c(O)c2)=O)C1 C=CC1CN(C(=O)CCc2cc(OC)ccc2OC)CC1NC(=O)C(CC)SC C(C)(CO)(C(C)(C)O)NC(CCC(C)NC(=O)CCOC1CCCC1)=O C1(NC(CSCCC(C)C)=O)CN(C(C2(C)CCCC2)=O)CC2(CC2)C1 C1(NC(C2C(OC)C2)=O)CCC(NC(=O)CC2CCN(CC(F)(F)F)C2)CC1 S(=O)(=O)(c1ccc(N2CCC=C(F)C2)c2cnccc12)NCC(C(C)(C)C)CO c1(-c2cc(CC)on2)ccc(CN2CCC(C(=O)Nc3nc(C)c(Cl)s3)C2)cc1 c1(C(N2CC3C(NC(C(C(C)C)C(C)C)=O)(C3)C2)=O)cccc2c1CCC2=O N1(CC)CC(C(N2CCCC2c2nc(-c3ccc(Cl)nc3)no2)=O)C(C)(C)C1 N1(CC(=O)NC(=O)NCC=C)CCCC(NC(C2(C)CC=CCC2)=O)C1C C12(C(N3CC4(N(C(C(C)Cc5cnn(C)c5)=O)CC4)C3)=O)CCCCN1CCC2 c1(C(N2C(CNC(C(C)CO)=O)CCCC2)=O)ccc2c(c1)COC(=O)N2 CC1CCCc2c(C(N3CCOC(CCCNC(=O)CCC(F)F)C3)=O)cnn21 N1(C(CC(C)OC(C)=O)=O)CCC(O)CC1.c1(COCCCO)scnc1C c1(C(C)C)ncc(C(=O)NCC2CC(NC(=O)COCC3CCCO3)C2)[nH]1 N1(C(CS(CC)(=O)=O)=O)CCC2CCCC(C1)N2C(c1ccc(CO)cc1F)=O N1(C(C2(CC)CCCC2)=O)CCCN(C(=O)CCc2cnc(C)s2)C(CO)C1 Cc1nc(C)n(CC(=O)NCCC2CCN(C(c3cnc(Cl)s3)=O)C2)n1 c1(CN(C2CC2)CC2(Br)C(F)(F)C2)ccncc1-n1cccn1 c1(C(N(CC(C)NC(C2N(C(C)=O)CCOC2)=O)C)=O)cnnc2ccccc12 Cn1nccc1CC(=O)NCCC1CCC(NC(C2(CCF)CC2)=O)C1 C1(OC)CC2N(C1)C2=O.c1(CNC(=O)CC2(O)CCC2)csc(-c2ccsc2)n1 N1(C(C(C)OCCC=C)=O)CCC2C(CCN2C(C2(c3oncc3C)CC2)=O)C1 N1(C(Cc2ccc(C)nc2)=O)CCC(NC(C23CCC(C)(C2)OC3)=O)C(CO)C1 C1(C(=O)NC2CCCN(C(C3CC(F)C(=O)N3)=O)C2)CCc2ncnn2C1 Cc1cc[nH]c(=N)c1C(=O)N(C)CC1CCN(C(=O)CC2OCCC2(C)C)CC1 CCC(F)(F)C(C)(C)C(=O)NCC12CCC(CC1)N2C(c1csc(C(F)F)n1)=O c1(C(=O)NCCCCC2CCN(C(C3COC3)=O)CC2)coc2c1CSC2 c1(NC(C2C=CCN2C(c2cc([N+](=O)[O-])cs2)=O)=O)cccc2nccn12 N1(C(CCC=CC)=O)CCN(C(=O)CCCCN2CCCC2)C(CO)C1 N1(CC(N2CCCC(CNC(CC(C)C)=O)CC2)=O)CCCCCCC1=O O=C(C1=C(c2ccccc2)CCCC1)N1CC=C(CNC(C2(CF)CC2)=O)CC1 c1(OCC)ccc2c(c1)C(NCc1cc(-c3ccccc3)ns1)CCO2 Cc1c(C(N2CC(NC(c3cc[nH]n3)=O)CC3(CC3)C2)=O)[nH]c2c(C)cccc12 S(=O)(=O)(c1ccc(NCc2cc(C)sc2)cc1Cl)N(C)CCN(CC(F)(F)F)C c1(-c2cc(C)cc(O)c2)cn2cc(C(N3CCCC4CCCCC34)=O)ccc2n1 C1(CNC(C2N(CC)CC2)=O)CC2CCCC(C1)N2C(=O)CCOC O=C1NCC2CCN(C(NC3=CCCCCC3)=O)CC12 C1(C(=O)OC)C(F)(F)C12CC(NC(c1sc(C(C)(C)C)nc1C)=O)C2 CCC(CO)(C(=O)N1CC2CC1(C(=O)NC1CCC13CCCC3)C2)OC n1(CC(=O)N(C(C)CNC(c2ccnn2C2CCC2)=O)CC)cnc([N+](=O)[O-])c1 C1(CNC(C(C)CO)=O)CC2(C1)CN(C(=O)Cc1cc(Cl)cs1)C2 C(=O)(C(C1=CCC2CC2C1)C(F)(F)F)OC.C12CC(C(O)C1)n1nnnc1C2 CS(=O)(=O)CC(=O)NC(CO)C(=O)Nc1cncnc1O c1(C(=O)NC2(CNC(C(C(C)C)O)=O)CCCCC2)cc2n(c1)CCSC2 C1(NC(CC(C)(C)C(F)F)=O)CCCC12CCN(C(=O)CCC(F)(F)F)CC2 c1(OC)ccc(OC(F)F)c(C(C)NCCC2CCCC3CC23)c1 N1(C(Cc2c(OC)ccc(F)c2)=O)CC(C)CN(C(=O)COC2CCC2)C(C)C1 c1(C(=O)NCCNC(C2C(c3n(CC)cnn3)C2)=O)ccc(Br)cc1 c1(OC)ncc(C(N2CCCN(C(=O)C=CC(F)F)CC2)=O)c(C)n1 C(C)(C)(C(C)(C)C)NC(CC1C(NC(c2cn(CC=C)nc2)=O)CCC1)=O C(=O)(CC(C)C(F)F)NC1C2CN(C(c3cc(CSC)c(C)s3)=O)CC21 C1(CC)CC(CC(=O)NCC2CCC(NC(=O)CSC)CC2)CCO1 CC1CN(C(c2cc(F)c[nH]2)=O)CC1CNC(=O)CCCCc1ccccc1 N1(Cc2ccc(CC(=O)OC)cc2)CCCC(NC(c2c(C)csc2Cl)=O)CC1 C1(F)(CNC(CCCC)=O)CCN(C(c2ccoc2CC(=O)OC)=O)C1 CC1=C(C(=O)NCC2CCCN(C(c3ccc(C(C)=O)c(C)c3)=O)CC2)CCO1 Cc1cc(C(N2CC(NC(=O)CCCc3ccccn3)C(C)C2)=O)c(C)o1 C1(NC(C(C)CN(C)C(C2CC=CC(O)C2)=O)=O)CCOCC12CCC2 c1(C(=O)NCC2N(C(c3c(C)nc(O)[nH]3)=O)CC(O)C2)c(N)sc2ccccc12 C1(C(=O)NC2C(NC(c3n(CC)ccn3)=O)C2)CCc2nncn2CC1 C(N=c1[nH]c2c(c(=NCc3ccsc3Br)[nH]1)CCCC2)c1ccc(OC)cc1Br c1(C(=O)NC(CNC(CCCOCC)=O)C)cc(O)c2sccc2c1 CC1CC(OC(=O)Cn2ccc(Br)cc2=O)CCN1C(=O)OC(C)(C)C C12(NC(C=C(C)C3CC3)=O)CCCC1N(C(=O)CCC1CNC(=O)N1)CC2 N(C(=NCCOCC)NCC1(C)CCCOC1)CC(C1CCOCC1)CC C1(C(N2C(CNC(=O)Cn3cnnc3O)CC2)=O)CC2CC1CC2(F)F c1(NC2C3N(C(C4C(C)CC(=O)N4)=O)CC(CC3)C2)ncnc2scc(Br)c12 C1(CNC(c2ccc([N+](=O)[O-])s2)=O)C2CCC(C2)N1C(c1cc(C(F)F)no1)=O C(c1ccc(F)c(F)c1)=CC=CC(N1CC(NC(C(CC)(C)CC)=O)C2C1C2)=O c1(NC(C2(NC(CC3C(C)CCC3)=O)CC(O)C2)=O)cccc(N=[N+]=[N-])c1 N1(C(CCS(C)=O)=O)CCCC(O)(CNC(=O)CN2CCCC2=O)C1 c1(C(N2C(C)CCC(NC(=O)C3=CCCSC3)C2)=O)[nH]nc([N+](=O)[O-])c1Cl c1(COC)ccccc1C(=O)N(CCCOCCN(C)C(C1CC12CCC2)=O)C CC(c1ccccc1Cl)=CC(=O)NC1CCCC(NC(=O)CC2CCN(C)C2)C1 N1(C(C(COCC)C)=O)CCC2(C(=O)NCc3cnc(C)c(C)c3)CCCC12 c1(C(=O)OC)nc(Cl)[nH]c(=NCC2CN(C(=O)C(C)(C)SC)CCCO2)c1OC c1(C(=O)NCCC2(C(=O)NCC(CCOC)(C)O)CC2)c[nH]c(C#N)c1C c1(C(N(CC(C)(C)NC(Cc2c(C)nn(C)c2C)=O)C)=O)cccc2oncc12 C1(C(=O)Nc2n(C(C)C)ncc2)CN(C(=O)CC2CN(C(C)C)C2)CCS1 c1(C(C(=O)NC(CNC(CCC=CCC=C)=O)CO)(C)C)ccccc1C C(=O)(CCCN1CCCC1)NC(C(=O)N(C(CC)C)C)C1CCCC1 CCC(CC)CC(F)C(=O)N1CC(CF)(NC(=O)CCN2CCC2)C1 Cc1ccc2sc(CN(C(c3ccccc3)CCc3ccccc3)C=O)cc2c1 C1(NC(C(C)Oc2ccc(C)cc2)=O)CCN(C(C2COC(=O)N2)=O)CC(O)C1 c1(C(=O)NC(CC)(CNC(=O)C(c2ccccc2F)C)CC)cc(Cl)ncc1O c1(C(N(C(CNC(C=CSC)=O)C)C)=O)ccc2cc([N+](=O)[O-])ccc2n1 CC(COC(c1cccnc1-c1cc[nH]n1)=O)C(C)(C)C C=CCCCCCC(=O)N1CCC(C)C1CNC(=O)Cn1ncc(O)nc1=O S(=O)(=O)(c1ccc(NCC2CCOC(CC)C2)nc1)NC(CC)COC C=CCC(C(=O)N(CCCC)C)NC(C1CCC(=O)CC1)=O CC(C)CC(C)(CNC(=O)C(F)C1CCC1)NC(c1csc(Br)c1)=O C1(C(N(CC(O)CF)C)=O)CC2CC1CC2NC(C1CC2(C1)CC(O)C2)=O C(=O)(CC(CC)C(C)C)Nc1cccc(CNC(COCC#C)=O)c1 C1(CNCC(C)(C)OC)CCN(C)CC1c1cnn(C)c1 c1(C(N(C2CN(C(c3c(CC)cccc3)=O)C2)C)=O)ccc2c(C)[nH]nc2c1 N1(C(C(CSC)(C)C)=O)C2CCC1C(C)C(NC(c1sc3cncn3c1C)=O)C2 C1(C(N2CC(F)C(F)C2)C(=O)Nc2c(C)c(Cl)ccc2)CCC2COCCC2C1 c1(C(C(=O)NC2CC(C)(NC(C=C3CCC(C)C3)=O)C2)O)ccccc1F c1(C(N2CCC(C(C)(C)NC(=O)C(F)CC3CC3)C2)=O)cnc(C(F)(F)F)nc1 N#CC1CN(C(c2ccccc2N(F)F)=O)CC1NC(c1cc(Cl)ncc1Cl)=O CCC(C(=O)OC)NC(c1nc(CNC(=O)Cc2cccnc2)cs1)=O C(C(N=[N+]=[N-])C(=O)NC1CC(CCNC(C2(OC)CCCC2)=O)C1)OCC CCC(C)(C(=O)NC(CNC(=O)C(c1ccccc1OC#N)O)C(C)(C)C)OC c1(C(=O)OC)cc2ccccc2[nH]c1=NC1CC2(CCCCCC2)C1 c1(C(=O)NCC23CN(C(C#C)=O)C(C2)CO3)ccc(S(N)(=O)=O)o1 N1(C(c2c(C)nn(C)c2C)C(=O)NCCCSCC)CCN(C)C(C#N)C1 C1(CNC(C2(C(=O)OCC)CC2)=O)CCN(C(=O)CC2CC23CC3)C1 c1(OC)ncc(C(=O)NC2CCCN(C(c3ccnc(CO)c3)=O)C2)cc1C c1(-n2ncc(C(N3C(CC(=O)OC)CC3)=O)n2)ccc(Cl)cc1 n1(C(C)(C)C)cc(CN(CC2CC2)CC2CC2)nn1.C12CC(C1)C(=O)N2 O=C(C1=C2CCN=C2NC=C1)NCc1ccc(SC2CCCC2)cc1 N1(C(c2c(C)noc2)=O)CCCCC1C1CCN(C(C2(C)CCN(C)C2)=O)CC1 C1(C)(CC)CC(C(N2CC=CC2CNC(=O)CC2(CSC)CC2)=O)C1 Cn1c(-c2noc(CSCCCO)n2)cc2ccc(Br)cc12 C1(C(=O)NCC23C(CN(C(C4(CCCC)CCC4)=O)C2)C3)CS(=O)(=O)CC(=O)N1 C1(N(CC)CC)CCN(C2=NCC3(CC3)N2)CC1 C12(NC(CC(c3cccc(Cl)c3)C)=O)CC(CC1CO)C2 c1(C(=O)NCCC(CNC(C(C)OCCC#C)=O)O)ccc(C)n(C)c1=O C1(NC(=O)CC2OCCCO2)CCCCN(C(=O)CC2CC3CC3C2)C1 C1(CNC(=O)CCC(=O)N2CCOCC2)CC(C(=O)N2CCCCCC2)=NO1 Cc1nc2c(cc1C(=O)N(C1CCC(NC(=O)CC3CC3)C1)C)c(C)nn2C c1(C(N2CCC(C(C)NC(C(CSC)(C)C)=O)C2)=O)cc(Cl)c(N)cc1F C1(F)(C(=O)NC(CCC)(C)C)CCN(C(C2C3CCC(F)C23)=O)CC1 N1(C(c2nc(CC)sc2)=O)CCC2C(C1)CN2C(C1CN(C2CCCCC2)C1)=O C1(NC(=O)CCc2ccsc2Cl)CCN(C(c2ccc(CO)cc2)=O)C12CC2 C1(NC(C(C#C)(C)C)=O)CCCN(C(c2snc(Cl)c2Cl)=O)CC1F Fc1cccc(Cl)c1CCCNC1CC1C1CC1 C(C1(O)CCCc2ccccc21)NC(c1cccc(Br)c1Br)=O N(C(=NCCN1CCCC1)NC(C)Cc1ccc(C)cc1)CC1(C(CC)C)CC1 C1(C)(COC)CC(NC(c2cncc(OC)c2)=O)CN1C(=O)C(C)SC N1(C(Cc2c(CC)cccc2)=O)CC2CCC1CN2C(=O)CCCCCOCC N1(C(C(C#N)C2CC2)=O)CCC(C(=O)Nc2cccc(CO)c2)C(O)C1 C1(NC(c2c(CC)nn[nH]2)=O)CC(C)CN(C(c2cc(C)c(CC)s2)=O)C1 c1(CC(=O)NC2CN(C(c3nc(C)oc3C)=O)CC2O)c(O)ncnc1O C12(NC(C=C(CCC)C)=O)CCCC1CN(C(=O)Cc1ccc(Cl)cc1)C2 N1(C(c2cc(C(CC)C)no2)=O)CCN(C(c2cnn(CCF)c2)=O)CCC1C c1(CC(=O)N(CCN(C(C)C)C(C2CCC(=O)N2C)=O)C)cc(Cl)sc1Cl N1(C(C2C(CC)CCCC2)=O)CC=C(C(=O)N(CCC2CC2)CC2CC2)C1 Cc1cc(C(=O)NC(C)CCNC(C2CCCCN2C)=O)cc(=O)n1C c1(CC)conc1C(=O)NC(Cn1cccn1)C(=O)NC(C)CCF C1(COC)(CNC(C2(C)CS(=O)(=O)C2)=O)CCN(C(c2csc(C)c2N)=O)C1 c1(OCC(N)=O)ccccc1C(=O)NCC1(F)CC(NC(c2ccns2)=O)C1 c1(C(COC)NC(=O)C(O)C2(N)CC2)cc(Cl)cc(Br)c1 C1(C(=O)NC(CCNC(Cc2c(C)ncs2)=O)C(C)C)CC2(CCCCC2)C1 C(CC(C(=O)NC(CCO)C(F)F)NC(=O)CCc1cn(C)nn1)OCC C#CCCCCC(=O)NC1CN(C(=O)COC2(C)CCCC2)CCC1C C1(C(=O)NC2CC(C)(NC(c3ccc(SC)o3)=O)C2)CCC2(CCC2)C1 C1(OC2CN(C(CC=C=C)=O)C2)CN(C(=O)C(C)C(C)C)CCO1 N1(C(C(n2cc(-c3cc4ccccc4[nH]3)nn2)C)=O)CCOC2(CCCSC2)C1 c1(NC(CC2C(NCc3nc(C(=O)OC)sc3)CCC2)=O)ccc(Cl)c(C)c1 C1(NC(c2cc(C(F)(F)F)cs2)=O)COC2CN(C(c3cccc(O)n3)=O)CC12 c1(NC(c2n(C(C)(C)C)nnn2)c2cnc[nH]2)ccc(F)c(Cl)c1 c1(OC)cc(O)c(C(N2CC(NC(=O)COC(C)(C)C)CCC2C)=O)cc1OC CC1=C(C(=O)NC2CCN(C(C3(F)CC=CC3)=O)CCC2CO)CCC(C)(C)C1 C1(NC(C2(C(C)C)CC2)=O)CN(C(c2cc3n(c2)CCSC3)=O)C2(CCCC2)C1 N#CC12CCC(C(N3CC=CC(NC(c4cc5n(n4)CCC5)=O)C3)=O)(CC1)CC2 N1(C(C(COC)O)=O)CC(C2(NC(=O)C(C)Sc3ccccc3Cl)CC2)C1 c1(C(N(C2CCC(NC(C(COC)O)=O)CC2)C)=O)cc2c(F)c(F)ccc2s1 C1(NC(C(C=C)(C)C)=O)CN(C(=O)C(CC(C)C)N(C)C)CCC1O C(=O)(C(C)(O)C(C)c1ccccc1)NCC(C)(C)NC(c1ccc(C(C)C)s1)=O CP(C)(=O)c1ccc(C(=O)NCC2CN(C(C3(C(F)F)CCCCC3)=O)C2)nc1 Cc1c(C(=O)NCC2CN(C(C3CCC3C)=O)C(C)(C)C2)nc2sccn12 C1(C(=O)NCc2cc(C)ns2)CC(C)(C)CCN1C(=O)C1=CCC(C)CC1 Cc1ccc(C)c(C(=O)NCCC2(O)CCN(C(=O)C(O)C3CCCC3)C2)c1 CCCCCC(O)CNC(C1C=CC(NC(=O)C(C)(COC)CC)C1)=O C=CC1CN(C(c2ccc(NC(C)=O)s2)=O)CC1NC(=O)CC1CCN(C)CC1 n1(CC)c(C(=O)NCCCNC(=O)CN2CSCCSC2)cnc1O Cc1c(C(=O)NC2CC3C(NC(c4cnn(C5CCC5)n4)=O)C3C2)cnn1C C1(NC(CCC(=O)NCC)=O)C2CCC(C2)C1C(=O)N(CCC(C)C)CCO c1(NC(N(CCCNc2nccs2)CCOC)=O)ccncc1 n1(CC)cc(CNC(N2CCC(c3nccn3C)C2)=O)nn1 CC1(C)C(NC(c2cnc(S)[nH]2)=O)CC1CNC(c1cc[nH]c1C1CC1)=O C1(C(=O)NCCC(C)N2CCC2)CC2(CCN1C(c1cnnn1C)=O)CC2 N1(C(CNS(NC)(=O)=O)=O)CCC(F)(F)C(CNC(=O)C(C(C)C)N(C)C)C1 N1(CC(=O)N(C(C(=O)NCc2ccc(Cl)o2)C2CC2)C)CCNC1=O c1(SC)nc(C(N2CCCC2C2C(CNC(=O)C(F)C(C)C)C2)=O)c2ccccn12 CCCCCCC(=O)NCC1C2CC2CN1C(c1ccnc(C)c1C)=O c1(C(=O)NCC2CN(C(COCCCC)=O)C3C2C3)cn2cnnc2cn1 C1(F)(C(N2CCC(OCC(=O)NC3CCCN(CCC)C3)C2)=O)CCN(C)CC1 c1(OC)ccc(Cl)c(C(=O)NCCC2CCCN(C(=O)C(O)P(C)(C)=O)C2)n1 C12(CNC(c3cc(CC)ncc3)=O)CC(CO1)N(C(c1nc(C)ncc1Cl)=O)C2 C1(C(=O)NCC(CC=C)NC(c2ncoc2CC)=O)CCCCN1CC(F)F C=CC(CC)CC(=O)NCCCN(C(=O)CC1(C(=O)OCC)CC1)CC CS(=O)C1CN(C(=O)CC2CCN2C(c2ccon2)=O)C1 C1(CC)CN(C(C2(O)CCOCC2)=O)CC1C(=O)N(CCO)CCN(C)C c1(C(=O)NCC2CC(COC)CN2C(c2cc(C)sn2)=O)ccc(O)cc1Cl C(=O)(C(O)CNC(C1(C)CCOC1)=O)N(CC#C)CC c1(C(N2CCCC(NC(C(CC)n3cccn3)=O)C2C)=O)cccc2nc[nH]c12 C1(NC(c2c(C)[nH]nc2C(C)C)=O)CCC2CC1CN2C(c1cc(CO)on1)=O C1(C(N2CCCN(C(c3cc(C#N)sc3)=O)CC2)=O)CCc2nnc(O)n2C1 C1(NC(c2scc(C)c2)=O)COCCN(C(=O)C(C)C(F)(F)F)C1 c1(OCC)ccc(C)nc1C(N1CC(C)(NC(=O)C=Cc2ccc(C)cc2)C1)=O c1(C(N2C(CCOC)CN(C(C3CCCS3)=O)CC2)=O)ncc2[nH]ncc2n1 c1(C(=O)NC2(C(=O)NCC(N3CCOCC3)=O)CCSC2)c(F)cncc1F C12(NC(Cc3nc(C)[nH]n3)=O)CCCC1N(C(c1cc(C3CCC3)on1)=O)CC2 C(=O)(C(F)C(F)(F)F)NC(CN(C(=O)C(C(C)(C)C)n1ccnn1)C)(C)C C(CC(=O)NC(C(=O)NOC1CCCC1)C1(O)CCC1)(C(C)(C)C)OC C1(C(=O)NC2CC(COC)C2)CCCCN(C(=O)CC(C)(C)C2CC2)C1 Cc1cncn1CC(=O)NCC(C1CCCCC1)NC(C12CC(C)C1C2)=O C1(NC(CN(C)C(N)=O)=O)CC(NC(=O)CCCCC2CC2)CC1O C1(NC(c2ncc(C)c(Br)c2)=O)CCC(O)CN(C(C2CCC2)=O)C1 N1(C(c2n(CCC)cnc2)C(=O)NC(C)(C)CC)CC(COC)CC1(C)C C(C1c2ccccc2CN1C(=O)C1=CCOCC1)NC(C(CC=C)C(C)C)=O C1(CNC(C(C)OC)C)CCCC12CCNCC2 C1(NC(C2C(C)(C(C)C)C2)=O)CCCC12CN(C(C1(CCN(C)C)CC1)=O)C2 N1(C(C2(OC)CCC2)=O)CCCC(C(=O)NC2CCC(N(C)C)CC2)C1 CCCCC(C)C(=O)N1CCCCC1C(N1CCCCC1CCCO)=O c1(C(=O)NCCOCCCNC(C(C2CCCO2)OC)=O)cnn(C)c1C C1(OC)CCN(CCCC2CCC2)CC1(C)OC c1(N(C(C)CCC2CCN2C(=O)OC(C)(C)C)C)cccc(C#N)c1 C1(C(N2CC(CC(C)NC(COC)=O)C2)=O)CC(OC)CC1OC C#CC1(C(=O)O)CCN(C(c2coc(SC)c2)=O)C1 C1(C(=O)NC(C)CCO)CN(C(=O)OC(C)(C)C)CC1C#N C1(C(=O)NC(CNC(C=COCC)=O)CCOC)(OC)CC(C)(C)C1 CC(C)C(CC(=O)NCCC1CCCCO1)NC(=O)CCCc1cncs1 C1(C(=O)NC2CC(NC(Cc3c(C)cccc3)=O)C2)CCCc2ccccc2C1 C1(CC(=O)NCc2cncc(C(N3C(C(=O)NC)C=CC3)=O)c2)NC(=O)NC1=O C(C(C)(C)CNC(=O)CC1CCCC1C)N(C(=O)CN(c1ncccn1)C)CC N1(C(C(C)(Cl)Cl)=O)CC2(CCCC(CNC(c3ccoc3Cl)=O)O2)C1 c1(C(=O)NCCC2N(C(C3C(CC(C)(C)C)C3)=O)CCCC2)cnc(N)c(Cl)c1 C(=O)(CS(=O)(=O)CC(C)C)NC(CC)(C)CNC(c1cnn(C(C)C)c1C)=O c1(C(C2(CCl)CCC2)NC(C)CC2CCC2)nnnn1CCCC1CC1 N1(C(c2snc(OC)c2Br)C(=O)NCc2ccco2)CCCC(C)(OC)CC1 C1(N(C(=O)C(CCC2CCC2)NC(=O)Cc2ccccc2)C)CCCN(O)C1=O CC(C)C(C(=O)N1CCC1CC1CC1)NC(=O)Cc1cn(C)nn1 C1(C)(CNC(CCCOCC)=O)CN(c2ccc(C(=O)OC)c(C)n2)CCO1 N1(C(C(C=C)C)=O)CCN(C(=O)C(c2cccc(C)c2)F)C(C)C1C c1(C(=O)NCC(CO)OC)cc(F)ncc1NC(C1CC(O)CN1C(C)=O)=O N1(C(C2(c3ccsn3)CC2)=O)CCC2C1CCCN2C(C1CC(C(F)(F)F)C1)=O Cc1cc(C(=O)NCC(C)CN(C(=O)CC(C)C)C)cnc1C(F)F N1(C(c2c(OC)scc2)=O)CC=C(CC(=O)N(C2CCC3CC23)C)CC1 C1(CC(=O)N(C)Cc2nc[nH]n2)(NC(C(COC(C)=O)C)=O)CCCCC1 c1(C(=O)NC2CC(CNC(C=Cc3nnn(C)n3)=O)C2)cccc2oc(=N)[nH]c12 N1(C(C2CC(OC)(OC)C2)=O)C2CCC(C(=O)NC3(C(O)CO)CCC3)C1CC2 C1(C(=O)NC(COCC)C(=O)NC(C)C(C)(C)CO)CC2C=CC1C2 C#CCCC(C(=O)OC)NC(C1CC(O)CN1C(=O)CC1C=CCCC1)=O C=CC1OCCC1C(N1CCOCC1CNC(=O)Cc1sc(C)nc1C)=O c1(CC)ocnc1C(N1CC(C(C)NC(=O)C(C)c2ccon2)C1)=O N1(C(C2(CC)CCCCC2)=O)CC2CCCC(CNC(=O)Cn3nccn3)C2C1 c1(CC)cccc(C)c1NC(=O)CC(C)CNC(=O)NC C(=O)(C1=C(c2cnn(C)c2)N(CC(=O)O)C(=O)NC1c1cccc(I)c1)OCC c1(-c2cn(CC3N(C(c4ncc(Cl)s4)=O)CCC3)nn2)cccc(Cl)c1[N+](=O)[O-] N1(C(c2c(CC)noc2)=O)CC2CCC2(NC(=O)C(C)=C2CC2)C1 C1(NC(CCSCC)=O)CCN(C(=O)C(c2cccc(Cl)c2)CC)CC1C(N)=O C12(CNC(CC3ON=C(C)C3)=O)CN(C(=O)C=Cc3ccccn3)CC1CCO2 N1(C(=O)CCC2CC2)CCC2C1CCCN2C(c1ccn(-c2ccccc2)n1)=O N1(C(CC(COC)C)=O)CCC(CCNC(=O)C(C)=CCO)C(F)(F)CC1 C1(NC(C2CC(C#N)C2)=O)CCN(C(=O)COC2CCOCC2)C1C1CC1 C=CCC(CC(C)C)C(=O)N1CCN(C(=O)CNC(=O)CNC(C)=O)CC1CO C12(C(=O)NC(C(=O)NCc3cc(C(C)C)on3)CC3CCC3)CC1CNC2=O c1(C(C)NC(C(C2CC2)NC(c2c(C)csc2)=O)=O)ncc(F)cn1 CCC(CC(F)F)C(=O)NC(C)CCNC(=O)C=Cc1cocn1 C1(NC(=O)C(F)=CC2CC2)CC1C1CCN(C(c2cc3cccnc3[nH]2)=O)CC1 Cn1cc(C=CC(=O)NCC2(NC(C3CC3c3cccc(F)c3)=O)CC2)cn1 c1(COCC(=O)NCC2(F)CC(NC(C3(CC)CCCC3)=O)C2)ccnc(O)c1 n1(CCC#C)c(N2CCC(OC3CCOCC3)CC2)nnc1CCCS(C)(=O)=O CON1CCC(N(C(=O)C(C(C)CC)N(C)C(c2cc([N+](=O)[O-])c[nH]2)=O)C)CC1 C1(NC(N2CC(C(F)(F)F)CC(C)C2)=O)CN2CCCC2CO1 CCCCCC(=O)NCCOCC(N1CCC(OC2(C#N)CC2(C)C)CC1)=O C=C(C)CCC(=O)N(C)CC1CCCN1C(c1c(C)coc1-c1ccccc1)=O C1(CNC(CC=CCC)=O)CN(C(C2(CO)CCOCC2)=O)CCCO1 C=CC1COCC1NC(=O)CN(C(C1COCCC1C)=O)C(C)C C(=O)(C1=C(CCOC)N(CC2CC2)C(=S)NC1c1c(Br)sc(Br)c1C)OCC c1(CC)ccccc1NC(N1CCC(CNC(c2ccncn2)=O)CC1)=O c1(CC)oc(C(=O)NC2CCCC2CNC(=O)CCc2ccc(C)o2)cc1C CC1(CNC(C2CC2(F)F)=O)CCCC1NC(C1CC(O)C1)=O CC(C)(C)C(O)CN1CCC1.C1(OC(=O)C=CCCCC)(OC)CSC1 C(=O)(C(C(C)(C)O)NC(C1CC2(CCC2O)C1)=O)NC1CC(C#C)C1 C(=O)(CCCCC(C)(C)C)N(C)CC1CCC2CNCC12CCO c1(C(C(=O)NCC2C(NC(=O)C=CI)CCC2)O)ccc(F)cc1 c1(C(C(=O)NC2CCCN(C(CNC(C)=O)=O)C2)C)cc2ccccc2o1 O=C(CCS(=O)(=O)C(F)(F)F)NC1CC(NC(C2CC23CCS(=O)(=O)CC3)=O)C1 C1(C)(CNC(C#CC)=O)CCN(C(C2(S(C)(=O)=O)CC2)=O)CC1 CC1C(N=c2[nH]c(=NCC3(CO)CC3)[nH]c3c2COCC3)CCCN1C c1(-c2ncc(C(N3CC(O)(C(C)NC(C=CCOC)=O)C3)=O)s2)ccccc1C C#CCC(CC#C)C(=O)N1CCCC(CNC(=O)CCc2ccc(Cl)s2)C1 C1(CC=C)(C(=O)NCC2CC(NC(c3snnc3CC)=O)C2)CCOCC1 C1(C(=O)NCC2CN(C(C(C)CN(C)C)=O)CC2O)CCC([N+](=O)[O-])CC1 c1(C(C)C(=O)NCCC2CC(NC(=O)CCc3cscn3)C2)ccc(F)cc1 O=S(=O)(c1cnc2c(Br)csc2c1)NCC1CCC(N2CCOCC2)CC1 Cc1ccc(O)cc1NC(C1C=CCN(C(C2CCC2(F)F)=O)C1)=O C1(NC(C(C)=C(CC)C)=O)CC2CC(NC(c3c(N)ccc(F)c3C)=O)CC2C1 N1(C(C(C)OCC)=O)CCC(CO)(CNC(c2cnn(C)c2C2CC2)=O)C1 CCC(C)CC(C)C(=O)N(C1CCC2CN(C(C3CC(O)C3)=O)CC12)C c1(CC(=O)NC(C(C)NC(=O)C(C)C2CC2)C)ccc(Br)c([N+](=O)[O-])c1 C1(C(=O)OC)CCCC(CC(=O)NCCNC(c2cccn2C(C)C)=O)C1 c1(CNC(c2cc(C)[nH]n2)=O)nc(CNC(=O)CCN2CCC(F)C2)cc(O)n1 C1(C(=O)NCCC(C)(C)NC(C=C(C)C(F)F)=O)CCc2cnn(C)c2C1 C(=O)(C(C)(F)C(C)(C)F)NCC(C)(O)CNC(=O)C1=CCCCC1 Cc1nc(C=CC(=O)NC2CN(C(C3CCCC(C)(C)C3)=O)CC23CC3)[nH]c1C N1(C(CC(CC)O)=O)CCc2cccc(-c3cn(Cc4ccncn4)nn3)c21 c1(OC)ccc(C(=O)NCC2CCN(Cc3cnc(Cl)s3)C2)c(OC)c1 C12(C(=O)NCCNC(CC)=O)CC(CO)(CN1C(C1CCC(=O)NC1)=O)C2 c1(C(=O)NCC2(NC(c3nn(C)c(Cl)c3)=O)CCC2)cc2ccncc2c(O)n1 c1(C(=O)NCC(C)CN2CCCC2=O)ccc(Cl)c(C#N)n1 N1(C(C(C2CCCN(C(C3CCCCCC3)=O)C2)C)=O)CC2CCC1C(O)C2O c1(C(=O)NC(CCNC(C(C)OCC)=O)C)ccc2c(c1)COCO2 N1(C(CC)=O)CCC(C(=O)N(CC(C2CC2)OC)CC)CC1 N1(C(CCCc2nc(C)sc2)=O)CCC2CCC12CNC(=O)Cc1ccsc1 c1(CC)cn2c(n1)CC(C(=O)NC1CC(CNC(=O)C(C)=C3CC3)C1)CC2 n1(C(C=C)C)nc(-c2ccc(Br)cn2)nc1CCc1cncnc1 c1(N2CCC(C(C)CO)CC2)cccc(S(=O)(=O)N2CCC=C(Cl)C2)n1 N1(C(c2cc(CC)sn2)=O)CCOCC1CNC(c1cccc(C)c1)=O N1(C(C(C)OCOC)=O)CCC2(CC1)CC(C(=O)NCc1ccc(CO)o1)C2 c1(N(CC)CC)ccc(C(=O)NCC2CCNC(C)C2)c(O)c1 C1(NC(C=CC=CCC)=O)C2CC3C1C3C2C(=O)NCC1(O)CC2CCC1C2 c1(NC(C2CCN(C(CCCC#C)=O)C2(C)C)=O)cn(C)c(=O)cc1C c1(C(=O)NC(C2CCCN2C(=O)CCC2(C)CC2)C)cc(NC(N)=O)ccc1F c1(C(N(C2CCCCC2)CCNC(C(C)N(C(C)=O)C)=O)=O)occ2c1CCC2 c1(CCNC(C(n2cc(C(C)OCC)nn2)C)=O)cnccc1OC c1(C(=O)NC(C)CCNC(C2(CF)CC2)=O)cc(-c2cnn(C)c2)on1 C1(C(=O)NCCCNC(C2(C)CC(C)C2)=O)CCN(c2ccc(Br)cn2)CC1 c1(C(=O)NC(C(=O)N(CCCN(CC)CC)C)CC2CCC2)cn(C)cc1C N#Cc1ccc(CC(=O)NC2CC(NS(N)(=O)=O)C2)c(Br)c1 CC(C)C(C(C)NC(=O)Cn1cnc(C(F)(F)F)c1)NC(=O)C=CC(=O)N(C)C Cc1cc(C(F)(F)F)ccc1Cc1cc(F)c(Cl)cn1.N12CCOC(C1)CC2=O c1(OC)cc(NC2CCC(n3ccc(NC(=O)OC(C)(C)C)n3)C2)nc(OC)n1 N1(C(C(CSC)C)=O)CCN(C(=O)CN2CC=CC2)CC1c1cc(F)ccc1F c1(-c2cn(C(c3nnc(-c4ccc(C)cc4)o3)C)nn2)ccc(C)cc1C Cc1nnc2n1CC(C(=O)NC1CN(C(c3ccc(=O)n(CCF)n3)=O)C1)CC2 Cc1ccc2c(c1)C(C(=O)NC1CC(NC(c3cnc(C(N)=O)s3)=O)C1)C2 N1(C(C2CCC(CC)O2)=O)CCC2(CC2NC(c2cc(C)n(C)n2)=O)C1 C1(NC(c2c(CNC(C3C(C)(C)CO3)=O)cco2)=O)CCOCC1O CCC(C(=O)N1CCC(O)(CNC(c2nccc3[nH]ccc23)=O)C1)C(C)(C)CC C1(CNC(C(C2CC2)OCC)=O)COCCN(C(c2cc(Br)cn2C)=O)C1 CC1(C)CCCC(C)(CN2CC(NC(N)=O)C(O)C2)C1 N1(C(c2cc(C(N)=O)oc2)=O)CC2(CCCC2NC(c2cc(Cl)sc2Cl)=O)C1 n1(CCC)nccc1C(=O)NCC(C)(C)OCC(=O)N(C(C)CS(C)=O)C1CC1 CC12CN(C(=O)C=CBr)CC1(C)CN(C(C1CC3(CC3)C1)=O)C2 c1(C(C(=O)NCCC)N(CC=C)CC2CCS(=O)(=O)C2)ccc(C(F)F)cn1 C12(NC(CNC(=O)OC)=O)CCC(CNC(C3SCCC3C)=O)(CC1)OC2 CCCCCCC(CC)NC(=O)C(O)CNC(=O)C(C)(C)C(N)=O CC1CCC(NC(c2ncsc2C(F)(F)F)=O)CN1C(C1CC1C1CC1C)=O C1(C(N(CC(CNC(CC(C)SC)=O)O)C)=O)C2(CCC2)C12CCC2 C1(C(N(C)C)=O)COCCN1C(C1C2CC=CCC12)C(=O)NCC(F)F Cc1cc(C)n(C)c(=O)c1CNC(=O)N(CC(O)CC(F)(F)F)C c1(CC)cc(C(=O)NC2(CC(N3CCC(F)(CF)C3)=O)CC2)nn1C Cc1ccc(CN=C(NC2CC(C)C2)NC2CCOCC2)cc1C#N C1(C(C(=O)N(CC=C)C(C)C)C)CCN(C(=O)CC2CCOCC2)C1 c1(SC)ccc(C=CC(=O)NCC(O)CNC(=O)CC2C=CCCC2)s1 CCCC(CCCNC(c1cocc1Br)=O)NC(=O)C(C)(O)C(C)C N1(C(CNS(NC)(=O)=O)=O)CC(CCNC(C23CSCC2C3)=O)OC(C)C1 C(C(CCN=c1nc2scnc2c(N2CCC(=CBr)CC2)[nH]1)OC)OC CCCCC(CC)C(=O)N1CCCOC(CCNC(c2cscn2)=O)C1 CCCCC(CCCC)C(=O)NC1CC2CN(C(c3[nH]c(C)nc3C)=O)CC2C1 Cc1ccc2c(c1)C(Nc1nc3c(Br)cccn3n1)CC2 Cc1[nH]c(C(=O)NC(c2ccc(F)cc2)CNC(=O)C(C)C)c(C)c1C C(C(=O)N1CCC(C(F)F)(CNC(c2occc2F)=O)C1)(C(C)C)SCC c1(C(=O)NCC(CO)NC(C(=O)NC(C)C)=O)ccc2nnc(O)n2c1 C(C(F)(F)C(=O)OCC)NC(CC1CC(CNC(CCC#C)=O)C1)=O Cc1nc(C)c(CNC(=O)NCc2ccc(CF)cc2)nc1C C=CCC(C(=O)N1CCCCCC1)NC(c1cc(OC)cs1)=O C1(OC)CC2CCC(C1)N2C(C12CC1CN(C(=O)CCCn1ccnc1)C2)=O N(C(=NCCc1cccs1)NCC(N1CCCCC1)C)CCSC c1(C(N2CC(NC(C34CC=CC(C3)OC4)=O)C2)=O)noc2cc(Cl)ccc12 C1(CNC(c2nn(CC)c(O)c2)=O)CN(C(c2cn(C)cn2)=O)CC(C)(C)O1 C(N=c1[nH]c(=NCCCCCF)[nH]c2c(F)cccc12)C1OCC(C)(C)OC1 Cc1nn(C)c2sc(C(=O)NCC3CN(C(c4nc(Br)c[nH]4)=O)CCO3)cc12 c1(C(N2C(C(=O)NC(C(CC)CC)C)CC(O)C2)=O)nccc2[nH]ccc12 c1(C(=O)OC)cc(CNC(=O)Nc2noc3c2CCC3)cnc1O C1(C(N(C(=O)OCCOC(N(C)CC)=O)C)=O)CC1(C)C N1(C(COCc2onc(CC)n2)=O)CCCC12CCN(C(=O)Cc1cnns1)C2 c1(C(CN(C(c2ccc(C3CC3)o2)=O)C2CC2)NC)ccc(Cl)cc1Cl C1(F)(CNC(C(CSC)OC)=O)CCCN(C(=O)C(O)C2CCCC2)CC1 C12(C(=O)NC(CNC(CC(C(C)C)O)=O)CO)CCN(CC1)S(=O)(=O)C2 C1(CC(=O)NC(CNC(C(C)N(C(C)=O)C)=O)(C)CO)CCC2CC1C2(C)C N1(C(C2CCCCC(=O)N2)=O)CC2CCN(C(=O)Cc3cccnc3)CC2C1 c1(C(N2CCC(NC(c3cc(C)n(C)n3)=O)C(O)C2)=O)n[nH]c2c1CCSC2 c1(OC(C)C(=O)NCC2CC(NC(c3ccc(N)o3)=O)C2)cccc(Cl)c1 C(=O)(C(O)CCC(F)(F)F)NCC(CCNC(c1c(CC)cno1)=O)OC CCC(CNCC1CCN(OC(=O)OC(C)(C)C)C1C)(CC)N(C)C CCC(CC(C)C)C(=O)N1CCC(CCC(N2CCS(=N)(=O)CC2)=O)C1 Cc1ccc(C(c2nnnn2C2COC2)NC(c2ccccc2C)C)cc1F C=Cc1cnn(C)c1C(=O)NC1CCCCC1NC(=O)Cc1csc(NC=O)n1 C=C(C)C(CC(=O)NCCN(C1CCN(C)CC1)c1ncccn1)OCC n1(CC)nc(C(N2CCC(C)C2CNC(c2cc(COC)oc2C)=O)=O)cc1O c1(C(=O)NC)cccc(C(=O)NCC2CCCCN2C(c2ccsc2C)=O)n1 C(CCCCC(=O)NCC(C)(CC(C)C)NC(C1OCCCC1(C)C)=O)OCC C1(N(C(C=C(C)CCC(=O)NCC(C)(O)C2CCC2)=O)CCO)CCOCC1 c1(CC)nc(=NC(CNC(=O)C=Cc2cnccn2)C(C)C(C)C)s[nH]1 C1(C(=O)NC(C(=O)NCC(C)C)(C)C)CCC(=O)CC1C C#CCC(CC#C)C(=O)N1CCCC(N(CCO)C(c2c[nH]c(C(N)=O)c2)=O)C1 c1(C(=O)O)cc(CN2CC(O)CC2CNC(c2cc(F)ccc2Cl)=O)ccc1Cl N1(Cc2cccc(SC)c2)CCC2(CC1)CC(N(C)CCO)C2 Cn1ncc(C(=O)NCCC2CN(C(=O)CCN3C(=O)CCC3=O)C2)c1C1CC1 N1(C(C=COCC)=O)CCC(NC(=O)C=Cc2nnc(C(C)C)o2)CC1C1CC1 c1(NC2CCC(=O)NC2)nc(=NC2CC(Cl)(Cl)C2)[nH]c2ccsc12 CC1CC(NC(c2cccc(Cl)n2)=O)CN1C(=O)C(C1CCCCC1)O C1(CNC(=O)CSc2nncs2)CCC2(CCC2)C1NC(=O)C1=CCC1 O=C(CC1=CCCC1)N1CCN(C(C2CCC23CCCO3)=O)CC1 c1(OCC(C(N2CC(OC)(CNCC(=O)OC)C2)=O)C)ccc(CO)cc1 c1(SCC)cccnc1C(=O)NCC1C(C)CCN1C(=O)C(F)OC c1(C(=O)NCC2(NC(C(C)CN(C)C)=O)CCOC2)cc(O)ncn1 C1(NC(C(C)OCC=C)=O)CN(C(c2cc(C(C)(C)C)on2)=O)CC1C(F)(F)F C(=O)(C(C(C)F)NC(=O)OC(C)(C)C)NC(CCNC(C(CC)NC(C)=O)=O)C c1(CNC(CCOCCOC)=O)cc[nH]c1C(=O)NC(C)CC(=O)OC C1(NC(C2CC(NC(Cn3ccc(C)c3)=O)C2)=O)CC2C(O)C(O)CC12 c1(C(C)(C)C)ccc(C(=O)NC2COCC2CNC(C2CCC2)=O)s1 C1(C(=O)NCC2CC2Cl)CN(C(C23CC2CNC3=O)=O)CC12CCC2 N1(C(c2c(C)nc(C(F)(F)F)s2)=O)CCN(C(c2ncoc2C)=O)CC(O)C1 N1(CC)CCOC(C(=O)NC2(C)CC(NC(=O)CC3COCCO3)C2)C1 Cc1ccc(C)c2[nH]c(C(=O)NCCN(C(C3CC3c3ccco3)=O)CC)cc12 N1(C(C(C)OC(C)=O)=O)CCC2(CC(NC(c3ncoc3C(C)(C)C)=O)C2)C1 C(=O)(C1CCc2ccccc21)NCC(CNC(C1CC(=O)OC1)=O)F c1(CC)cc(C(=O)NC2CCCCC2NC(=O)C=C(C)Cl)nn1-c1ccccc1 CC1CCCCN1CC(=O)NCC1(O)CCN(C(=O)CCNC(N)=O)C1 C1(C(C)NC(=O)CC2CC2(C)C)CCCCN1C(=O)CCc1cnco1 N1(C(C=C=C(C)C)=O)CCN(C(=O)C=C2CCN(C)CC2)CC(C)C1 C1(NC(CC)=O)CCCC12CN(C(c1ccccc1C(F)F)=O)C2 N1(C(C2CCCC2(F)F)=O)CCC(C)(C(=O)NC2(C(N(C(C)C)C)=O)CC2)C1 N1(C(COC)=O)CC(NC(C2(CSC)CC2)=O)C(NC(CCOC(C)C)=O)C1 C(CCCCCNC(c1ccc(=N)[nH]n1)=O)N(C(C1(C(=O)OCC)CC1)=O)C N1(C(C(C(C)C)OC(C)=O)=O)CCC2CN(S(=O)(=O)CC(C)C)CC2C1 C1(C(=O)NC(Cc2cc(C)[nH]n2)C)CCOCCN1C(=O)COCCC(C)C c1(C(N2CCCC(N(C(C(F)=CCC)=O)CCOC)C2)=O)ccnc(Cl)c1N C#CC(C(C)C)NC(=O)C(Cc1ccoc1)NC(c1cnn(CC)c1)=O c1(OCCCC)ccc(C(=O)NC2CC2NC(c2scnc2Cl)=O)cc1Cl c1(SCC(=O)NC2(CNC(C(C)n3cccc3)=O)CCOC2)ccccc1O C(C(C)(C(C)C)NC(c1cn(C2CCCC2)nn1)=O)NC(c1c(SC)snn1)=O c1(Nc2ccc(OC)cc2OC(F)F)ccnc2ncc(Br)cc12 c1(CCCC)nc(C(=O)NCC2(NC(c3ccc(CO)o3)=O)CC2)cs1 CC(C(=O)N1CC(NC(=O)CN(C)C(N)=O)C(CC(C)(C)C)C1)C(C)(C)C C12(C(N(C3CCCC3)CC=C)=O)CC(CN1C(C1C3CCCC13)=O)C2 C1(NC(C(CC)O)=O)CN(C(c2cc(C)c[nH]2)=O)CC1n1ccnn1 c1(OC)ccnc(-c2cccc(CN3CCC(n4ccnc4)C3)c2)n1 N1(C(CC(CC)CN(C)C)=O)CCCC(N=c2cc(C)[nH]c(C(C)C)n2)(CO)C1 c1(C(N2CCC(C)C(NC(=O)C(C)(C)F)C2C)=O)c(F)cccc1[N+](=O)[O-] n1(CC(=O)NC2CC2NC(C2CCCC2O)=O)nnc(C2CC2)n1 CCCN=c1[nH]c2c(c(=NC3CC(=C4CCC4)C3)[nH]1)COC2 C=CCC(C(=O)NCC1CC1CC(=O)NC1CS(=O)(=O)C1)C(C)C C(=O)(C1=C(F)CN(C(=O)CC(O)CC(C)(C)C)CC1)N1CC(NC(C)=O)C1 C(=O)(C(CCC1CCC1)NC(C1CN(C)CCO1)=O)NCc1c(C)ncs1 C(=O)(C1CCCc2nn[nH]c21)N(CCN(C(C(CC=C)C)=O)C)C C1(C(=O)NCC2CCCN2C(=O)Cn2cc(CO)nn2)CCN(c2nccs2)CC1 N(C(=NCCF)NCC(=C1CCOCC1)Br)CC(=C)F N1(C(C(N)=O)=O)CC2C3CCC(C(NC(c4cnnc(O)c4)=O)C3)C2C1 C=C1CC(C(=O)NCCn2cnc(C(=O)NCCS(N)(=O)=O)c2)(COC)C1 c1(COCC)nc(C(C)Sc2cnn(C)c2)n(-c2cnnn2C)n1 CCCCCC(O)C(C)C(=O)NCCC1CCN(C(=O)CCC2CCCC2)C1 c1(C(=O)NCC(N(C(C2CC(CC)(CC)C2)=O)C)C2CC2)cnn(C)c1CC c1(CC(C)C)ccc(C(C)C(N2CC(NC(=O)CSC3CC3)C(SC)C2)=O)cc1 Cc1cc(F)c(C(=O)NC2CCC2NC(=O)CC2C=NN(C)C2=O)c(Br)c1 c1(C(CC(C)C)NC(c2[nH]cc(C(C)=O)c2C)=O)nnc2ccccn12 CCC(C)(C(=O)N1CCC(C(C)(C)C)(CNC(c2c[nH]c(=N)o2)=O)C1)C(N)=O c1(C(=O)NCC2CC2c2cc(C)on2)nccnc1O c1(C(N2CC(C)C(CCNC(=O)CC3CCCN3C)C2)=O)ccc(P(C)(C)=O)o1 C(N=c1[nH]c(=NC2CCC(=O)NC2C)c2cc(F)cc(F)c2[nH]1)c1cnc(C)[nH]1 C1(NC(CNC(=O)OC)=O)CCN(C(c2ccc(C3CC3)cc2)=O)C2(CCC2)C1 C1(C(=O)NC(C2CN(C(c3cccnc3F)=O)C2)C)CNC(=O)N1C CCC(CC(F)(F)F)C(=O)N1CC(NC(c2c(C)ccnc2C)=O)C(N=[N+]=[N-])C1 c1(C(N2CCCCC(N(C(=O)CCS(C)=O)C)C2)=O)cnc2c(F)cccn12 c1(C(C)NC(=O)NC(CC(C)(C)C)c2ccc(F)cc2)ccc2c(c1)OCO2 C(=O)(C(C)(C)CC(F)F)NCCC1(CNC(C2(CC(C)C)CCNC2=O)=O)CC1 N(C(=NCCCCl)NC1CCCC(n2cccn2)C1)CC(=O)OCC1CC1 C1(NC(CCC)=O)CCC(F)(CNC(c2ccc(I)cc2)=O)C1 c1(NC(C2C(NC(CCc3ccc(OC)cc3)=O)C2)=O)cccc(OC)c1C#N c1(OC(C)C(=O)N(C)CCN(C(=O)CN2CCC(C)(O)C2)C)cccc(F)c1 C1(C(=O)NCC(CC)(C)OC)CCC2(CC2)N1C(=O)CCCc1cnn[nH]1 Cc1ccc(N)c(C(N2CCC(NC(=O)CSCc3cccnc3)C2)=O)c1F c1(N2C(C)CC(CNC(Cc3c(OC)ccc(C)c3)=O)C2)nc(C)ccc1C#N CC1(C)CCC(C(N2CC(O)CC2CNC(c2nccc(Cl)c2O)=O)=O)CC1 c1(C(=O)NC(CCN(C(C(CC)(C)OC)=O)C)C(C)C)cccc(F)c1C(C)C C1(CNC2(c3nnnn3C)C(CS(N)(=O)=O)CC2)CCS(=O)(=O)CC1 C1(C(N2C(CNC(C3(C#C)CCC3)=O)COCC2)=O)CNC(=O)CC1(C)C c1(C(=O)OC(C)C(=O)NCc2cncn2C)cc(N2CCOCC2)c(Br)cn1 c1(CCC(N2C(C)C(NC(=O)Cc3ccoc3)CC2)=O)ccc(S(N)(=O)=O)cc1 c1(C(C)C)cccc(C(=O)NC(c2ccnn2C)C(N2CCCCC2)=O)c1 CC1CC(C(=O)NCC(N2CCC2CC(=O)NCC2CCC2)=O)CCS1 c1(C(C)(C)C(=O)NCC(C2CCOCC2)O)cc(F)ccc1Br N1(CC)CCC2(CC1)CC2C(N1CCC(C(=O)N(C2(C)CCS(=O)(=O)C2)C)C1)=O N1(C(c2cnc(-c3cccs3)o2)=O)CCN(C(=O)CSC2CC2)C(CC2CC2)C1 c1(C(=O)NCC2C=CCN2C(C2CC2c2ccccc2)=O)cc2scnc2[nH]1 c1(CC(=O)N(CCS(CC)=O)c2ccccc2)c[nH]c2cc(F)ccc12 C1(CNC(CC(C(C)C)O)=O)CN(C(=O)COCCOCCO)C2(CCC2)C1 CN1CCC(C)(C(=O)N(CCC(=O)NC2(C)CC3CC3C2)CCO)C1 O=C1CN(C(=O)NCc2ccco2)c2ccc(O)cc2N1 Cn1nc2c(c1N)CN(c1nc(N3CCC(CF)C3)nc3c1SCC3)CC2 C1(OC)CC(C(=O)NC2(COc3ccccc3)COC2)N(c2cc(C)ncn2)C1 c1(C(N2CC3CC2CN3C(c2nc3cnccc3s2)=O)=O)nccc2occc12 N1(C(CC2CC(C)(C)OC2)=O)Cc2ccnn2CC(NC(=O)CN2CCCC2)C1 c1(-c2cccc(N3CCC(NC(CC)=O)CC3)c2)ccc(C#N)c(Cl)c1 CC(C)C(C)C(C)CC(=O)N1CC(CC(C)NC(c2ccc(Cl)cc2Cl)=O)C1 c1(C(N2CCN(C(c3c(CC)csc3)=O)C(C)C2)=O)cnc2n1CCCC2C Cc1ccccc1C=CC(N1CC(N(C)C(c2cc(C(C)C)ccc2F)=O)C1)=O N1(CCC)CC(C(N2CC(CNC(=O)C=Cc3ccco3)(OC)C2)=O)CC1=O CC1CCN(CCC(=O)NCC2(C(C)(F)F)CC2)CC1 c1(C(N2CCC(C(C)NC(CC3ON=C(C)C3)=O)CC2)=O)cc(C#N)c(C)cn1 O=S(=O)(c1c[nH]ccc1=NC1CC2(CCC2)C1O)NC1CC(F)(F)C1 Cc1noc(CCC(=O)NCCC2(NC(c3cc(C(C)C)[nH]n3)=O)CC2)n1 C#CCCC(C(=O)NC1CC1CC)NC(c1cccc(CC)c1)=O C(CCSC)(C(=O)NC(C)CN(C(=O)Cc1nnc(-c2ccccc2)o1)C)OC n1(CCCCO)nc(CCC(F)(F)F)nc1-c1ccc(C2CCOCC2)cc1 N1(C(CSCC#C)=O)CCC(NC(=O)CCOCCN(C)C)CC(C)(C)C1 N1(CC)CCCC1C1CCCN1C(C)=O.n12nnc(c1C(F)(F)F)NCC2 n1(C2(CCN3CC(OCC)C3)CC2)cc(CNC(c2cc(C(F)(F)F)cs2)=O)nn1 C12(C(=O)NCC(c3cccc(Cl)c3)NC(CC(C)C3CC3)=O)CC(CCO1)C2 C1(NC(c2n(C)cc(Cl)c2)=O)CCN(C(c2csc(C3CC3)n2)=O)CC1CO CCC(C)(C)NC(C)C(=O)N(C(C)C(=O)N(CC(C)C)C1CC1)C C(CC(C)N=c1nc(N2CCCC(C(C)(C)C)CC2)c2c([nH]1)CCCC2)SCC S(=O)(=O)(c1ccc(N2CCC(OC)CC2)c(C#N)c1)NCC(C(CC)C)O N1(Cc2ncc(C)nc2)CCC2(CC2C(=O)NCC2CCN(C)CC2)C1 C(=O)(C1=CCOCC1)N(C1CN(C(=O)C(c2cscn2)N(C)C)C1)C CC(C)CC(CNCCCN(C(Cc1ccccc1)C(=O)O)C)c1ccccc1 c1(NC(C2(C)CN(C(c3c(CC)cccc3CC)=O)C2)=O)ccc(Cl)c(C#N)n1 c1(N2CCC(OC(C)C)CC2)nc(NC2COC3(CCC3)C2)c2cnn(C)c2n1 C=CC1OCCCC1C(=O)NC1(c2ccccc2)CC(NC(=O)CN2CC=CC2)C1 c1(C(N(CCN2CCN(C(C3CCC(C)S3)=O)CC2)C)=O)cccc2cnsc12 Cc1coc(C(=O)N(CC(C)O)CCNC(C2CC(C)(C)O2)=O)c1 Cc1ccc(Cl)c(C(N2CC(NC(=O)CCC3(C)CC3)C3CC23)=O)c1 C1(C(=O)NCC2(CNC(C(CC)OC)=O)CC2)CC2(CCCCC2)C1 Cc1nn(C)c(C)c1C(=O)C(=O)NC1CN(C(C23CCC2C3)=O)C1 Cc1c(NC(C2CN(C(C3CC4CCC3O4)=O)CCC2O)=O)cccc1F C1(CCNC(c2cncc(C)c2)=O)CCN(C(c2[nH]c(O)nc2C)=O)C(C)C1 C1(NC(C(C)C2CCCC2)=O)CC2(C1)CC2NC(c1cnccn1)=O c1(NC(CC2C=CC(NC(CN3CCC(CC)C3)=O)C2)=O)cn(CC)nc1C#N c1(OCCC)ccc(C(=O)NCC2(CNC(C3(C(C)C)CC3)=O)CCC2)cc1 C1(CC)CCN(C(c2cccc(C)n2)=O)C1CNC(=O)C(=O)NC(C)C C12(CNC(CCC=C(C)C)=O)CC1CN(C(c1cnn(C(C)C)c1C(F)(F)F)=O)C2 C1(c2nnnn2C2CCCC2)(NCCc2ncc(Cl)cn2)CCCSCC1 N1(C(C2(C)CC2C(F)(F)F)=O)CCN(C(C2CN(CC(F)(F)F)C2)=O)C1 c1(C(N(COCC)CC)=O)cc2c(OC)c(OC)ccc2[nH]1 C(=O)(CCS(=O)(=O)c1ccccc1)N1C(CNC(CC(C=C)C)=O)C(O)C(O)C1 c1(C(=O)NC2C=CC(CNC(C3N(C)CCC3)=O)C2)cc(C2CC2)ccc1Cl C(=O)(C1=C(C)N(C)c2ncnn2C1)N1C2(CN(C(COCCC)=O)C2)CCCC1 C12CC(C1(C)C)CC(=O)NCC=CC(=O)N2.C(C(CO)OC)N(C)CC C1(NC(C(c2ccc(F)cc2)CC)=O)CC2CC1N(C(c1scnc1C)=O)C2 N1(C(c2c(COC)cccc2)=O)CCCC(NC(c2sc(C)cc2Cl)=O)CC1 c1(C(N2CCC(CCCNC(C(C)SC)=O)CC2)=O)sc2ncccc2c1N c1(CC)cc(C(=O)NC2CCCC2CNC(C2(C)CS(=O)(=O)C2)=O)n(C)n1 C1(CCNC(CC=C)=O)CN(C(C2CC2OC(C)(C)C)=O)CCO1 C12(C(=O)NCC3C=CC(NC(C(n4c(C)ccn4)C)=O)C3)CCC(CO)(CC1)C2 C1(CNC(C(CC#C)C)=O)CCN(C(c2cc(C3CCC3)no2)=O)C1(C)C N#Cc1csc(CNC(=O)CNC(=O)C(O)C2CCC2)n1 C(=O)(C(C(=O)NCC(C)(O)CNC(C1(c2ncco2)CC1)=O)C1CC1)OC C(=O)(C1CCCc2nncn21)N1CC2N(C(C3(CC#C)CCC3)=O)C(CC2)CC1 C1(O)(C(C)NC(C(CC)C)=O)CCN(C(=O)CCSc2nccn2C)CC1 CC(C)CC(C(=O)NCC(CO)NC(c1cn(C2CCOC2)nn1)=O)C(C)C c1(NC2C(CNC(CC(COC)(C)O)=O)CCCC2)ncnc2c1cnn2CC CC1(C)CCN(C(C2CC(=O)N(O)C2)=O)CC1CNC(=O)Cc1cncnc1O c1(C(=O)OC)cn(C)nc1C(=O)NC1CN(C(=O)CN2CCC(C)C2)CC1C N1(C(c2ccc(COC)o2)=O)CC(NC(C2CC3CCC3C2)=O)CC12CCCC2 N1(C(CNC(C2C(C)C2)=O)=O)CCC(NC(=O)CCOc2ccccc2)CC1C c1(-c2nn(-c3cccc(C(N)=O)c3)c(CSC3CCC3)n2)cc(F)c(N)c(F)c1 N1(C(c2cc(CC)[nH]n2)=O)CCC12CN(C(C1COC(=O)O1)=O)C2 c1(C(=O)NC2CN(C(C3=CCCC3C)=O)CC2C)n[nH]c2c1CCCC2 CC1CN(C(C2(c3ccnc(Cl)c3)CC2)=O)CC1CCNC(=O)Cn1cnnc1 c1(C(C)OC)ncc(C(=O)NC(C)CC(C)NC(=O)CSc2ccccn2)s1 Cc1ccc(C(=O)NCCCCCCNC(=O)CC(C)N2CCCC2=O)cc1Cl C(=O)(C(C=C)SC)N(CC(CC)NC(COCCC=C)=O)C1CC1 n1(CC(=O)N(CCNC(C2CCS(=O)(=O)C2)=O)CC)ccc2ccccc12 c1(-c2nnc(N(C)Cc3cnc(C)s3)n2CC2CC2)cncc2c(F)cccc12 Cc1cc(NC(c2ncccc2NC(=O)CCC(C)C)=O)n(CCO)n1 C=CC1(O)CCN(C(C2CCC(CNC(C3(C#N)CC3(C)C)=O)O2)=O)C1 C(C1c2ccsc2CCN1C(C1(C)CCC1)=O)NC(C(C)c1cc[nH]n1)=O c1(C(C)C)ccc(C(N2CC(CNC(C3(C)CCNC3=O)=O)CC2C)=O)cc1Cl C1(C(=O)NCc2cnns2)(NC(=O)CC2CCOC2)CCCC1 N#Cc1cccc(C(N2CC3C(C2)N3C(=O)COC2CCCC2)C2CC2)c1 C(C(C)(C)CC(=O)NCc1ccccc1C)NC(C=C(C)C(C)C)=O N12CC3CCCC3(C1)C(=O)N(CCCO)CC2=O.NC(=O)CSC1CC1 C=CC(CCC)CC(=O)NCC1(O)CCCN(C(=O)C=Cc2cn[nH]c2)C1 Cn1c(CNC(=O)Cn2cc(CNC(=O)C(=O)NC3CC3)nn2)nnc1O Cc1cc(NC(=O)CN(C2CCC2)C(C2CCN(C)C2)=O)c(O)c(C)c1 C1(O)(NC(c2ncccc2Cl)C2CC2)CCCN(C(N(c2ccccc2)C)=O)C1 C1(CNC(c2c(CC)nc(C)nc2)=O)CN(C(=O)CCC#N)CCC12CCC2 c1(C(N(C)CCC2CCCCN2C(=O)CC2CC3CC3C2)=O)cncc(F)c1Cl c1(C(=O)NC2CC(C)N(C(=O)CN3CCS(=O)(=O)CC3)C2)cnn2c1CCCC2 C1(NC(=O)CC2CC2)CC1C1CCN(C(=O)Cc2cc(F)ccc2O)CC1 N1(C(c2ncn(C(C)C)n2)=O)CCC(CCNC(=O)COc2ccsc2)CC1 c1(CC(=O)N(C)CCNC(=O)CCCn2cncn2)ccc(Cl)nc1 c1(C(N(C(c2ccccc2)CNC(C2C(=C)C2)=O)C)=O)cc(Cl)c(Cl)c(Cl)c1 C1(NC(c2c(O)ccc(C)c2)=O)CC(NC(c2coc(Cl)n2)=O)C12CCOCC2 C1(CC(=O)NCCC(=C)CNC(c2cncc(C(F)(F)F)c2)=O)CCNC(=O)C1 c1(C(N2CC(NC(c3cncnc3)=O)C(F)C2)=O)n[nH]cc1[N+](=O)[O-] N1(C(CN(C(=O)OC)C)=O)CCC(NC(C2CCCN2N=O)=O)C1(C)C C(c1ccc(F)cc1)=C(C)C(=O)OC1CC2CC(C(=O)OC(C)(C)C)C2C1 C1(C(N2CCCC(O)(C(C)C)C2)=O)CCN(C(=O)CC2CCOC2=O)O1 c1(CNC(C(F)=C(C)C)=O)ccc(CNC(C2COC(C(F)F)C2)=O)cc1 Cc1cc2[nH]c(C(=O)NC3CCCN(C(C4CN(C)CCO4)=O)CC3)cc2o1 Cc1nc(C(=O)NC(c2ccccc2)C(N2CCOCC2C)=O)ccc1F c1(C(=O)NCC(CNC(c2cc(C)[nH]n2)=O)C)ccnc(-n2cccn2)c1 CC(CSC(F)(F)F)C(=O)N1CC(C(N)=O)(CNC(=O)C(C)(C)NS(C)(=O)=O)C1 c1(C(N(CC(O)CNC(=O)Cc2ccccc2)C)=O)ccc(CCO)cc1 CCC(CC(F)(F)F)C(=O)NC(CCN(C(=O)C(CC)CC)C)C(C)(C)C c1(OC)cc(C(=O)NC(C2CCN(C(=O)C3=CCSC3)C2)(C)C)ccc1O c1(C(=O)NC2CCN(Cc3ccc(O)cc3F)C2)c(F)ccc(Cl)c1Cl C1(C(N2CC(OC)C(NC(c3csc([N+](=O)[O-])c3)=O)C2)=O)CCc2nc(C)cn2C1 Cc1cnc(Cl)c(C(=O)NC(C2CN(C(c3cccn3C(C)C)=O)CCO2)C)c1 c1(CNC2C=CC(C(=O)NC3CC(=O)OC3)C2)ccc(Cl)c(Nc2ccncc2O)c1 CC1(CCNC(c2conc2CNC(c2cscn2)=O)=O)CCCO1 N1(C(C(CC2CCC2)OC)=O)CCC2(CC(C(=O)NCCC3CCCOC3)C2)C1 C(=O)(C(F)(F)C(O)C1CC1)N1CC(CN2CCN(C(CC(C)O)=O)CC2)C1 C1(NC(CCC(=O)NCCC)=O)CN(C(=O)CCCn2ccnc2)CC1N=[N+]=[N-] c1(C(=O)NCC2C(NC(C(C3CCC3)OCC)=O)CC2)ccc2nccnc2c1 C(=O)(C(C1=Cc2ccc(OC)cc2OC1)N1CC(OC)C(CO)(OC)C1)NCC(=C)C C#Cc1cccc(CC(=O)N(CCCNC(=O)C=CC=CC)C)c1 CN1CCCC1C=CC(=O)NCCNC(=O)CN(C1CCSC1)C c1(C(N(CCNC(C=C=C(C)C)=O)C)=O)cc(F)c(N)cc1F C(=O)(NNC(=O)C(C)SC1CCCC1)c1cc(OC)c(C(C)(C)C)cc1 Cc1ccc(C)c(CNC(=O)C(CO)NC(C2CC2(F)Cl)=O)n1 C=Cn1ccnc1C(c1nnnn1CCSC)NCC(c1ccc(F)cc1)(C)C c1(C(=O)NC(C(C)NC(C2CC(CC)C2)=O)C)ccc(N2CCCC2)cc1 c1(C(=O)NCC(c2cccc(OC)c2)O)ccc([N+](=O)[O-])c(OC(F)F)c1 C1(C(C)NC(C2(COC)CCCC2)=O)CCCN(C(c2nn(C)nc2C)=O)C1 N1(C(c2c(OC)ccs2)=O)CCCC(C)(C)C1CNC(C1(S(C)(=O)=O)CC1)=O C12(NC(c3cn(CCCC)nn3)=O)CCC1CN(C(C1(C)C(C)(C)C1(C)C)=O)C2 c1(C(=O)NC2C(OC)CN(C(C3(O)CC3(C)C)=O)C2)nn(C)cc1S(C)(=O)=O C1(C(C)C)CCc2sc(C(N3CCC(C)C3CNC(=O)C(C)N(C)C)=O)cc2C1 Cn1ncc2cc(-c3nc(NC(c4ccc([N+](=O)[O-])cc4Br)=O)cs3)ccc12 Cc1cc(C(=O)NC2CCCC2C(=O)NC(C)Cc2cccnc2)cnn1 N1(C(C(=O)NC2(C)CC2)C2CC2(Br)Br)CCn2c(cnc2C(F)F)C1 CC1CC(NC(=O)Cc2cc[nH]n2)CCN1C(=O)Cn1cccnc1=O N1(C(C=C(CC)C)=O)C2CCC1C(F)C(NC(=O)Cc1c(Br)cnn1C)C2 c1(OCC(=O)NC2CC(CN(C(C(C)OC)=O)C3CC3)C2)cccc2ccccc12 C=CC(C)C(=O)N(C(CNC(=O)CCc1cnn(C)n1)CC)C c1(C(=O)NCCC(=C)CNC(=O)C(n2nccc2C)C)ccc(O)cn1 C1(CC(=O)N(CCF)CC)CCN(C(C2C3CCC(F)C23)=O)C1(C)C c1(C(N(CCNC(C2CNC(=O)N2)=O)CC2CC2)=O)ccc2oc(=O)oc2c1 N1(C(CC2CC(OC)C2)=O)CCN(C(c2cccc(-n3cncn3)c2)=O)C2CC12 C=CC1CCCC(NC(C2(C)CCCN2C(=O)CCCCCOC)=O)C1 O=C1CCC(CC(=O)NC2(C(=O)NCCC3COCC3O)CC2)CN1 N1(C(c2cnc(CC)nc2C)=O)CC2CC(NC(=O)C(C)(C)C(N)=O)C(C2)C1 C(=O)(CN=c1[nH]cnc2ccc([N+](=O)[O-])cc12)N1CCCc2ccccc2C1.CCC CC1(CC(=O)NC2(C3CC3)CC2)CCN(C(=O)CN2CCOC2=O)C1 C1(C(=O)NCCCCCCNC(c2nnn(C)c2N)=O)CC2(CO1)CC(F)(F)C2 N1(C(c2c[nH]c(Br)c2)=O)CCC2(CCN(C(=O)CC(O)c3ccccc3)C2)C1 c1(C(C)C(=O)NC2CCN(C(C3CCC(C)(C)C3)=O)CC2)ccc2c(c1)OCO2 C1(NC(CC(=O)NCC#C)=O)CCN(C(=O)CC2C=CS(=O)(=O)C2)C12CCCC2 c1(CN(C)CCNC(c2nn(-c3cccc(Cl)c3)cc2O)=O)ccc(C#N)cc1 N1(C(c2cn(C)nc2)=O)CC(O)(C2CCN(C(C3(Cl)CC3(C)C)=O)CC2)C1 N1(CC(=O)NC)CCCCC(NC(=O)C(N2CCC(C)C(O)C2)=O)C1=O C1(C2CN(C(c3cnc(C(C)(C)C)nc3)=O)C2)(NC(CCC#C)=O)CC1 c1(COC)ccccc1C(=O)NCCCN(C(C1CCC(C)CC1)=O)C(C)C n1(CCS(N)(=O)=O)nc(CC2CCC2)nc1-c1cnn(CC(F)F)c1 C1(NC(Cc2c(C)nsc2)=O)CC(CNC(=O)CN(C2CCC2)C)C12CCC2 C1(N(C(=O)COCC2CC3(CC3)C2)C)CCCN(C(C2CCOC2)=O)CC1 N1(C(C(C)NC(CC)=O)=O)C2CCCC1CN(C(=O)C(O)CC(C)C)C2 CN1CC=C(CC(=O)N2CC3CCC2(CNC(c2cn(C)cn2)=O)CC3)CC1 N1(C(c2cc(CN(C)C)on2)=O)CCC(O)(CCNC(C2(C)COC2)=O)CC1 c1(OC)cccc2c1OC(C(=O)NCCC1(NC(c3coc(CO)c3)=O)CC1)C2 C1(CCC(=O)NCCCSCC)CCCCN(C(=O)CCCOC(C)C)C1 C(CC(C(C)C)NC(=O)CCC(C)NC(c1cnc(OC)s1)=O)OC Cc1nc2c(s1)CCCC2C(=O)NCCC(O)CNC(C1CCCCC1)=O C(=O)(C(C#N)C(C)(C)C)N1CCC(C(CO)NC(C2(CC)CCCCO2)=O)CC1 C1(CC(=O)NCC2CC(NC(C3CCN(C(CC)=O)C3)=O)C2)CCCC12CC2 c1(C(=O)OCC)ccc(-c2nc(CCN=[N+]=[N-])no2)s1 C=C1CC2(C1)CC(C(=O)N(CC(C)N(C(=O)CCN1CCC(C)CC1)C)C)C2 C(=O)(C(C)(CC(F)(F)F)OC)NCCN(C(=O)CN(C)C1CC1)CC C(=O)(CCCCCC1NC(=O)NC1)NCC1(F)CCN(C(C2CCC(C(N)=O)C2)=O)C1 c1(OC)cc(CN2CCOCC(NC(c3cnc(Br)s3)=O)C2)ccc1I c1(C(C2CCCOC2)C)cn(CC2CCCN2C(C2(F)CCOC2)=O)nn1 C1(N(C(C2CCN(C(=O)C(C)(C)CCOC)CC2)=O)CC)CC(C(C)(C)C)=NO1 CC(C)CS(=O)(=O)N1CCN(CCNC2(CF)CCNC2)CC1 C(CN=c1ccnc(C2CCC2)[nH]1)N(C(c1cn(-c2ccccc2)cn1)=O)CC CC1COCC(C(=O)NCc2c[nH]nc2C(=O)NCC2(C)CSC2)O1 c1(C(=O)Nc2cccc(NC(C3CCC(C)(CC)O3)=O)c2)cc(Cl)ncc1O CCC(CCC(=O)NCC12CC(CC)(CN1C(=O)CC1CCSC1)C2)OC N1(C(C(=Cc2ccncc2)C)=O)CC2CCC1CC2NC(=O)Cn1nccn1 C(=O)(C1=NNC(=O)CC1)NC1CC(CNC(C2C(C)CCOC2)=O)C1 C1(NC(CCNC(=O)OCC)=O)CCC(CC(N2CC(C)(OCC)C2)=O)C1 S(=O)(=O)(c1oc2ccc(Cl)cc2c1C)Nc1c(C(=O)OC)cc(F)cc1 c1(C(=O)NCCOCCN(C(C(C)N(C)C)=O)C)cccc2c1S(=O)(=O)CCC2 c1(C(N2CCC(C)C2CNC(c2c[nH]nc2[N+](=O)[O-])=O)=O)cc(F)cc(N)c1F c1(C(=O)NCC=CCNC(C2OCCO2)=O)ccc2nc(O)nc(O)c2c1 CC1(O)CN(C(C2CCC(C3CC3)N2C(=O)CCCn2cncn2)=O)CCC1O c1(-c2c(F)ccc(OC)c2)cc(C(=O)NC(CO)C(C)O)c2cn[nH]c2c1 CC1(C)C(C(N2CCN(C3CCN(C(C4CC(F)C4)=O)C3)CC2)=O)CC1(F)F C1(NC(Cc2n(C)ncc2)=O)CC2(C1)CN(C(c1ccncc1Br)=O)C2 C1(C(=O)NC2CC(=C)C2)CC(C)CN1C(=O)CN1CCN(C)CC1 C(=O)(CCC(=O)c1cccs1)N1C(Cn2cc(CNC(C)=O)nn2)C=CC1 N1(C(C(C)C2(O)CCC2)=O)CC(O)CC1(C)C(=O)N(C)Cc1ccncn1 CC1(C)COC(CNC(=NCCF)NCc2ccc(F)cc2O)=N1 c1(CC(=O)NC2CC3CC(NC(c4cc(F)c[nH]4)=O)CC23)c[nH]c2ccccc12 N1(C(C=C2CCC(C)C2)=O)CCc2ccc(Cl)c(F)c2C1C C1(NC(C2(C)CN(C(CC(=O)NCC#C)=O)C2)=O)CCOC12CCCC2 C1(C(=O)NCCOC(CNC(c2c(C)cncc2)=O)(C)C)CC(C2CC2)=NO1 CCC(C#N)(CC)C(=O)NC(C)CNC(=O)CCc1ccc(F)nc1 C1(N(C(C(C)Cc2ccco2)=O)CCO)CCN(CCN(C)C)CC1 Nc1cc(C(N2CCC(NC(C3CCCCCC3)=O)C23CCC3)=O)cc(F)c1O c1(C(C)(C(=O)NCC(O)C(C)C)NC(CSC)=O)ccc(C(F)(F)F)cc1 N1(C(C=CCC)=O)CCc2cc(CNC(C3CC(OC)C3)=O)ccc2C1 S(=O)(=O)(c1cccc(C(=O)NCCCCNC(C2CC(=O)N(O)C2)=O)c1)NCC CCC(C)(CCO)NC(=O)CC1CCCN(C(=O)C2=C(Cl)CC2)C1 C(=O)(CCC(C)(F)F)NCC(CO)NC(C(CC)n1ccnc1)=O C1(C)(C(N(CCN(C(=O)CC2CC(C)(C)CO2)C)C)=O)CNC(=O)N1 c1(CNC(C2CCC(NC(CC(=O)OCC)=O)C2)=O)c(Cl)cccc1Cl C1(NC(c2[nH]cc(CC)n2)=O)CN(C(=O)C(n2ccc(C)n2)C)CCC1CO c1(C(N2CC(C)C(Nc3nc4cccc(F)c4s3)C2)=O)c(Cl)ccc2c[nH]nc12 CCS(=O)(=O)CC(=O)NCC1(CNC(=O)CCN(C)CCO)CC1(F)F C1(C(=O)NCC(CCOCC)NC(C2(CC)CCCCC2)=O)CCS(=O)(=O)N1 C1(C(=O)OC)CC(F)CN1C(C1CC2CC2N1C(C12CC(C(F)(F)F)(C1)C2)=O)=O CCCCC(CC(=O)NCC1CC(O)(CO)C1)NC(=O)C(C)(C)Cl c1(C(N2C(CNC(C3N(C)CCC3)=O)CC(C)(C)C2)=O)ccc2n[nH]cc2c1 N1(C(C=Cc2n(CC)ccn2)=O)CCC(C2(NC(c3nnc(S)n3C)=O)CC2)C1 N(C(=NCc1nn(C)c2ccccc12)N1CCC(C2CCCC2)C1)C(CC)C N1(C(c2cc(COC)no2)=O)CCOCC(NC(c2ccc(O)nc2C)=O)C1 C1(NC(C2CSCCO2)=O)C=CC(CC(N2CCCC2CC2CC2)=O)C1 c1(C(=O)NCCC2(OC)CN(C(c3cncc(C)c3)=O)C2)cccc(SC)c1 C1(=CC(=O)N(C(CN(C(C(=Cc2ccco2)C)=O)C)C)C)CCC(C)CC1 N1(C(CCc2cn(C)nc2)=O)C(C(=O)NCCC2=CCCCC2)CCC12CC2 Cc1nc2c(C)csc2c(=NCC(C)NC(=O)COc2c(F)cccc2F)[nH]1 c1(CSC)noc(CCC(=O)N(C)CC2CCN(C(C3CC(Cl)(Cl)C3)=O)C2)n1 c1(C(N(CC(CN(C(=O)CP(C)(C)=O)C)O)C)=O)ccc(C(F)(F)F)nc1O C1(OC(c2cc(C3CCNC3)[nH]n2)=O)CNC(=O)C(F)(F)C1 c1(N(C(N(C(C2CCCO2)C)C)=O)Cc2ccccn2)ccccc1F C(=O)(C#CC1CC1)NCc1c(CCNC(CN(CCC#C)C)=O)ocn1 N1(C(C2CCN(C)C2)=O)CCC2(CCN(C(c3cscc3C3CC3)=O)C2)C1 CC(C)C(C(=O)NC1CC1CNC(=O)CC1CCCC1)c1cccnc1 c1(C(=O)OC2CCN(CCCCC)CC2)ccc2ccc(OC)c(OC)c2n1 c1(CN2CCC(F)(C(=O)NCCC3CCCCC3)C2)ccc(O)cc1O c1(C(=O)NC2CC(C)N(C(=O)Cc3ccncc3)C2)cccc2ccsc12 CC1(CO)CCCN(N2CCC(NC(c3cccc(C(F)(F)F)c3)=O)C2)C1 CC1CCN(C(c2ccc(Cl)cc2)=O)C1C(N1CC(C)(c2ccccc2)C1)=O c1(N(C(N2CCC(O)C2C)=O)CC)cccc2cccnc12 C1(CNC(CCC2(NC(C(C)OCC3CC3)=O)CCC2)=O)CCC(C)(C)O1 N1(C(C(C(C)C)F)=O)CC2(C(=O)NC(C)C(F)(F)F)CC1CO2 N1(C(Cc2cc(C)sc2)=O)CC(F)(F)CC1CNC(=O)COc1cn[nH]c1 CN1CCC(C)(C(N2CCCC(C(=O)NC3CC(F)(F)C3)C2)=O)CC1 C(=O)(CC1=CCN(C)CC1)NC1C(CO)CCN(C(c2c(C)ccn2C)=O)C1 c1(CN(CC(O)Cc2nn[nH]n2)CC)ccc2c(c1)OCO2 C1(NC(CCC(=C)Cl)=O)CC2(CCCCN2C(=O)Cc2cc(C)on2)C1 C(c1cn(C)cn1)=CC(=O)NCC1(OC)CN(C(=O)CCC2CCCC(O)C2)C1 c1(C(=O)NC(C2CCN(C(c3ccno3)=O)CC2)(C)C)cc2c([nH]1)CCC2 Cc1nn2cc(C(=O)NC3CCCC3NC(c3ncoc3C)=O)nc2s1 N1(C(c2cnn(CC)c2Br)=O)CC(NC(=O)C(C)P(C)(C)=O)CC(O)C1 C1(C(=O)NCC2C3CN(C(c4cc(CCO)on4)=O)CC23)CCC2(CCC2)CO1 N1(c2c(OC)cncn2)CC=C(CCNC(=O)C(C)Sc2ccccc2)CC1 Cc1cc(C(=O)NC(C)C(=O)NCc2sccc2C)ccc1O C=CC1(NC(=O)C(CCC)NC(=O)C(n2ccc(C)n2)C)CCCCC1 N1(C(c2scc(C)c2)=O)CC2CCCC(C1)N2C(=O)C(F)C(F)(F)F C12(CNC(CCCCC=CC)=O)CN(C(=O)C(C)(CO)NC(C)=O)CC1CCO2 CC1(C)CC(CC(=O)N(C(=O)CN2CC(c3ccncn3)C2)C2CC2)NC1=O c1(C(=O)NCC2CN(C(c3cc(C)c(F)nc3)=O)C(C)C2)cccc([N+](=O)[O-])c1 C1(C(=O)NCC2(C(N(CC(C3CCC3)OC)C)=O)CCCO2)CCC(C)CC1 Cn1ncc(C(=O)NCc2ccc(C(N3CC4CCC4(CO)C3)=O)cc2)c1C#N Cc1cc2ccc(C(=O)N(CC(C)CNC(C3(CF)CCC3)=O)C)cn2c1 N(C1CC(C)(C)Cc2oc(C)cc21)C(C(CC)NC(=O)CN1CCN(C)CC1)=O c1(NC(N)=O)cccc(C(=O)NC2CN(C(=O)CCc3cc(Cl)no3)C2)c1 C1(NC(CCOCCCOC)=O)CC12CCN(C(c1c(C)cccc1F)=O)CC2 CN1CC(C)(C(=O)NCC(O)C(=O)NC2CCOCC2F)CC1=O C1(CC=C)(NC(c2cn(C(C)C)nc2C)=O)CCN(C(=O)CSCCOC)C1 C1(C(C(=O)NCc2cscn2)F)CCN(C(=O)Cn2ccnc2)C1 N1(C(c2c(NC)cncc2)=O)CC2COCC2(C(=O)NC2C3CCCOC23)C1 c1(-n2ccc(C(=O)OCC)n2)cc(F)ccc1F.c12cnn(c1)CCS2 Cc1cnc(CN2CC(CC(=O)Nc3ccnc(-c4ccncc4)c3)C2)c(F)c1 c1(C(=O)NC2CN(C(C3CC3(Cl)Cl)=O)CC(F)(F)C2)ccc2c(c1)OCCN2 N1(C(Cc2ccc(SC)cc2)=O)CCCC(N(C)C(c2ccnc(F)c2)=O)CC1 c1(C(=O)NCC(C2CCCN(C(c3cnc(C)[nH]3)=O)C2)C)cnc2[nH]cnc2c1 c1(C(=O)NC(C2N(C(C(F)=CC)=O)CCC2)C)ccc(N(C(C)C)CC)cc1 C1(c2n(CC)nnn2)(NCc2cc(C)ccc2OC)CCN2CCCCC12 c1(C(N2CCC(NC(=O)C3=CCCS3)(CF)C2)=O)cccc2[nH]ccc12 Cc1nc(C)c(C(=O)NCC2(O)CC(NC(C3CC3C(C)C)=O)C2)[nH]1 CC(CC(F)F)C(=O)N1CCCC1CNC(=O)C(C)(C)c1ccns1 C1(C(=O)NC(CNC(CCC(=C)Cl)=O)(C)CC)CC12CCCCCC2 c1(C(N(CCC(C)NC(C2(CCCC)CC2)=O)C)=O)cccc2c1NCC2 N1(CC)C(=O)CCC1C(=O)NCC(C)CN(C(=O)C(C1(O)CCCC1)F)C C(C(=O)NC1COCC1CNC(=O)CC#N)(C(C)(C)C)SC c1(C(=O)NC2CN(C(CCC(C)SC)=O)CC(O)C2)ccc2c(c1)C(C)(C)CO2 c1(NC(=O)NC(CCC)C(=O)N(C)C)ncccc1C#N C1(N(C(=O)Cn2ccc(C3CC3)n2)CC)CCCN(C(C2(O)CCC2)=O)C1 C(C(CC(F)(F)F)NC(c1ccnn1C)=O)NC(C(C)OC)=O N1(C(CC(C2CC2)NC(c2cccc(CC)c2)=O)=O)CCCCCCC1C N1(CC)CC(C(=O)NC(C(=O)NC(c2cncnc2)C)C2CC2)CC1=O N1(C(c2cccc(Cl)c2F)C(=O)NCC(=C)C)C2CCCC1CC1(CCC1)C2 C1(CNC(C(CC)n2ccnc2)=O)CN(c2cc(OC)ncn2)CCCO1 C1(C(N(C(C)C)CCN(C)Cc2cc(Cl)sc2Cl)=O)CC2CC2CC1C N1(C(CC2(C)CC2)=O)CCN(C2CCC(NC(=O)CC3CC(C(N)=O)C3)CC2)CC1 C1(C(=O)NCC(CO)NC(c2cc(C)cc(O)n2)=O)Cc2cccc(C)c2O1 C(CC(F)F)(C(=O)NCc1cnccc1C)NC(COCCC=C)=O C1(C(C)C(=O)NC2CCCC2NC(c2coc(C(N)=O)c2)=O)CCS(=O)(=O)CC1 N(C1CCc2ccccc21)C(C1CCCN(C(=O)C(=O)NCC(F)F)CC1)=O Cc1c(N)ccc(C(=O)NC2CC(C)N(C(c3cnnn3C)=O)C2)c1F N1(C(C(CC)CC)=O)CCC(C)(C)C1CNC(C1CCCC(C(N)=O)C1)=O N1(C(CCCC=C)=O)CCC2(CCN(C(c3cccc(C(=O)N(C)C)c3)=O)C2)C1 n1(CC(C)C)cccc(C(N2CC3CC(NC(c4cn(C)nn4)=O)C2C3)=O)c1=O CC1C(NC(c2ccc[n+]([O-])c2)=O)CC2CCC1N2C(c1cn(C)nn1)=O C=C(C)CCCC(=O)NC1COCCN(C(C2(CF)CC2(F)F)=O)C1 c1(C(=O)NC2C3CN(C(C(=O)NC4CC4)=O)C2C3)ccc2nc(Cl)nn2c1 N1(C(c2n(CC)cc(Cl)c2)=O)CCC(NC(=O)C(C)Oc2ccccc2)C(F)C1 C1(CC(N2CCC(NC(CC(C)CN(C)C)=O)CC2)=O)CC2(CCOCC2)CO1 C1(NC(c2cnn(CC3CC3)c2)=O)CC2(C1)CC2C(N1CCC1CC1CCC1)=O N1(C(C2(C)COC2)=O)CCC2COC(CC(=O)NC3CC(n4ccnn4)C3)C2C1 N1(C(c2c(F)ccc(C)c2)=O)CC(NC(=O)C(F)CC2CCCC2)CC12CCC2 C(=O)(C1=CC2CC(C1)CC2O)NCC(C)NC(c1cc(C)c(C)s1)=O N1(C(CC(C)c2ccco2)=O)CCCN(C(=O)CC2COC3CC2C3)CC1C CC1=NOC(C(=O)NC2(C)CC(NC(c3conc3C(C)(C)C)=O)C2)C1 C1(N(C)C(c2ccns2)=O)(CC)CN(C(=O)CC2(OC)CC2)C1 C(=O)(C1=CCCN(C(=O)C(CO)OC)C1)N(CC=C)CCO C1(NC(C2CC(CN(C)C)C2)=O)CCCCN(C(C2CC(=O)CCO2)=O)C1 c1(C(N2CCC(CNC(C(CC)C)=O)C2)=O)cc(Cl)cc(C)c1OC Cc1[nH]nc(C(N2CCC(Cc3ccncc3)C2)C(=O)NC2CCOC2)c1Br N1(C(CCCCC#C)=O)C2CC=C(C(=O)N3CCC3=Cc3ccccc3)C1CC2 c1(OCC)ccc(C)c(C(=O)NCC#CCNC(=O)CCNc2scnc2C)c1 CCCC(C(=O)NCC1C2CN(C(=O)CSCc3cccc(C)c3)CC12)C(C)C c1(NC2CCCC(NC(C=Cc3ccc(C)o3)=O)C2)ncnc2c1c(Br)nn2C c1(C(=O)NC2CCCN(C(C3C(C)OCCC3)=O)C2)c(F)ccc(F)c1N C1(C(=O)NCC(C)(C)N2CCCC2)CC(NC(=O)CC2CCCCC2O)C(O)C1 C(=O)(C(F)(F)C(F)(F)F)N.c1(COC2CCN(C(C=C(C)Cl)=O)C2)ccnc(S)c1 N1(C(CN(C)C(=O)C2CC2)=O)CCC2(CCCN2C(=O)CC2CCS(=O)(=O)C2)C1 N1(C(Cc2cc(OC)no2)=O)CCCCCC(NC(c2ccc(F)cc2O)=O)C1 C(C(C)C(C)C(=O)NCCOC1CN(C(c2ccc(=O)n(CCF)n2)=O)C1)OC c1(C(N2CC(NC(C(COC)O)=O)C(C(F)(F)F)CC2)=O)c(F)cc(Cl)cc1F C(c1cnc(O)nc1O)=CC(=O)N(C1CCCN(C(c2cnn(C)c2F)=O)C1)C N1(C(c2cc(C)oc2)=O)CC(C)(C)CCC1CNC(c1conc1C1CC1)=O CP(C)(=O)CC(=O)NCC1(NC(=O)CC(O)C2CCCC2)CCCC1 c1(C(N(CC(CNC(C(C(=O)OCC)(C)F)=O)(C)C)CC)=O)cnc2ccccn12 c1(NC(C2CC(F)CN2Cc2ccc(Cl)nn2)=O)ccc2nonc2c1 c1(C(N2CCCC2CN2CCCS2(=O)=O)C)cc2cc(Br)ccc2[nH]1 C1(NC(c2ccc(CC)o2)=O)CC(NCC=O)C12CCC2.C1CNC(=O)N1.CC c1(OC)ncc(Br)c(=NCC2CCCC2NC(c2ccc3c(c2)C(C)CO3)=O)[nH]1 c1(OC)cc(C(N2CCOC(CC(=O)Nc3ncc(F)cc3O)C2)=O)cnc1I c1(NC(N2CCCc3cc(Br)ccc32)=O)cnc2c(c1)C(=O)NCC2 C1(C(=O)NC2C(CC(=O)NCC(C=C)O)CCCC2)CCCC2(CC2)C1 N1(C(=O)OC(C)(C)C)CC(C2CC2)(C(N2CCN(c3cccc(O)n3)CC2)=O)C1 C1(N(C(CC=CCC)=O)C)CCCC(NC(c2cnc(N(C)C)cn2)=O)C1 C12(NC(C(C)SCCCC)=O)CCC(C(=O)NCC3CCC(C)(C)CO3)(CC1)C2 CC1(C)CCN(C(N2CCC(C)(F)C2)=O)C1NC(=O)C(F)(F)F N1(C(C=CCC)=O)CCCC1C1CCCN1C(c1nc(CC)oc1C)=O C(=O)(CC(C)(C)C(F)F)N(C)CC1OCCN(C(C(F)=C(C)C)=O)C1 n1(CC(N2CC(CNC(C(C)=CC)=O)CC2(C)C)=O)cc(C#N)c(O)nc1=O C(=O)(C(CC)(CC)CC)N(CCN(C(=O)C=Cc1cc[nH]n1)CC)CC n1(CCC=C)cc(C(=O)NCC2CCCN2C(=O)CCCOCCC)nn1 N1(C(c2nc(CC)[nH]n2)=O)CCC(CO)C(NC(=O)C=C2CCCCC2)C1 C1(NC(CC(C)NC(N)=O)=O)CN(C(c2cccc(C3(C#N)CC3)c2)=O)CC1O C=CC1(CC(=O)NCc2cc(Cl)no2)CN(C(=O)C=Cc2cscn2)C1 Cc1cc(NC(C2(F)CCN(C(c3cncc(Br)c3)=O)C2)=O)c(Cl)cc1Cl C1(NC(C(C)CC2CCCC2)=O)(CO)CCCN(C(C2(C(F)F)CCCC2)=O)C1 CC1=C(C(=O)N2CCC(C(C)NC(c3cnnc(Cl)c3)=O)C2)CCO1 Cc1cc(C(=O)NC2CCCC(NC(=O)COCC(C)C)C2)cc2c1CCC2 c1(CN(C(=O)C(C)(CC)N(C)C)C)cc(I)ccc1Br c1(C(=O)NC2(C(=O)OC)CC23CCC3)cc(Br)cc(Br)c1 Cc1c(NC(C2CC(O)CN2C(=O)C(C)(C)O)=O)cccc1CO C1(C(N2CC(CCNC(C(C)(C)OCC)=O)OCC2)=O)CS(=O)(=O)CC12CCC2 C1(NC(c2n(CC)ncc2Cl)=O)Cc2ccccc2C1NC(=O)C=C(C)C(C)C CN1CC=C(CC(=O)NC2CCCC2NC(c2cnc(Cl)cc2N)=O)CC1 CCCCCC(O)C(=O)N1CC(C(O)C(=O)NC2CCC(C)(C)CC2)C1 C1(CC(=O)NC2CCOCC2NC(=O)Cc2c[nH]nc2O)CCC(F)(F)CO1 Cc1cc(C(N2CCC(NC(=O)C=Cc3c[nH]nc3C)C23CC3)=O)c(C)c(C)c1 c1(N2CCC(C(=O)NCC(c3nccc(C)c3)O)CC2)ncnc2oc(C)nc12 c1(CNC(C2CCCO2)=O)n[nH]cc1C(=O)NC(c1cccnc1)CO CC1CN(C(=O)CN(C)C)CC(C)C1NC(=O)CS(=O)(=O)Cc1cccs1 CCCCC(O)C(C)C(=O)N1CC(C2CC2C(N2CC(C)(OC)C2)=O)C1 N1(C(C(CCCC)C)=O)CC(NC(=O)CNC(=O)NC2CC2)CC2(CC2)C1 C(=O)(C#CC1CCOCC1)NC1CC(CNC(c2ccc(SC)cc2)=O)C1(C)C N1(C(c2nc(C(C)(C)C)oc2)=O)CC2(CCN(C(c3ccc(Cl)nc3N)=O)C2)C1 c1(C(=O)NC2CC(N(C)C(C3(N4CCCCC4=O)CC3)=O)C2)ccc(F)c(Cl)c1 C1(NC(C2CCC(=C3CCC3)CC2)=O)CN(C(c2ccc(CO)cc2)=O)C2CC12 c1(N2C(CCC)SCC2)cc(S(=O)(=O)NC2CC2CCC)ccc1C#N C1(NC(c2c(OC(C)C)n[nH]c2)=O)CCCN(C(c2ccnn2C(C)C)=O)C1C C=CCC(CC(C)C)C(=O)N1CC2(C1)CN(C(=O)CCCn1c(O)nnc1O)C2 C1(C(=O)OCC)CC(NC(=O)CC2(C(=O)OCC)CCC2)CC1C(=O)OC(C)(C)C C(CCN(C)C(c1c[nH]nc1C(C)(C)C)=O)(C(C)(C)C)NC(C(CC#C)C)=O C1(COC)CN(C(c2ncc(N)cc2Cl)=O)CCN1C(=O)C(C)OCC(C)C C1(NC(c2n[nH]c(C)c2C)=O)CC2CCC(C1)N2Cc1cccn2ccnc12 C12(C(=O)NCCCN(C(C3C4CC4C4CC34)=O)C3CC3)CCN(CC1)C2 N1(C(COC(C)C)=O)CCCC(NC(c2c[nH]nc2-c2ccco2)=O)C1C c1(OCC(=O)NC(c2nccn2C)C)ccc(F)cc1.C12CC1CNC2=O NC1CCC2CCN(C(=O)NC3CC4OC(=O)CC34)C12 NS(=O)(=O)c1n[nH]cc1C(=O)NCCCC1CCN(C(C2CCCC2O)=O)CC1 Cc1c(C(=O)N(C)CC2(NC(C3CCCCC3O)=O)CC2)cc(F)cc1Br Cc1nc(C2CC2)ncc1C(=O)N(CCn1cc(CCCS(N)(=O)=O)nn1)CCO C1(C(=O)NC(CC=C)CNC(C2(c3ccnn3C)CC2)=O)CCC(N(C)C)CC1 c1(NC(C2(OC)CN(C(C(CCC)O)=O)C2)=O)nc(OC)ccc1[N+](=O)[O-] C1(CC)CCCC(CNC(C2CCOC2CNC(c2cnc(S)nc2)=O)=O)C1 C1(NC(c2csc(CO)n2)=O)CN(C(=O)C=CC2CCCC2)C2(CCCOC2)C1 c1(C(N2CCCCC2CSS(C)(=O)=O)C(=O)NCC(C)C)ccc(C#N)cn1 C1(NC(=O)NC(C)CCO)CCN(c2cnccn2)CC1 C1(CC(N2CCC(C)(CNC(c3c[nH]c(C#N)c3)=O)C2)=O)COC2(CCC2)CO1 c1(C(=O)NCC(C)NC(C(C)NC(C)=O)=O)cnn(-c2ccccn2)c1 Cc1ccc(O)c(C(N2CC=CC2C(=O)NCC(=O)NCC(F)F)=O)c1 C1(NC(CNS(CC)(=O)=O)=O)COCCN(C(c2cnc(Cl)c(Cl)c2)=O)C1 c1(C(=O)NCC(CC(=O)NC(C#C)CC(C)(C)C)C)ccn2nccc2c1 c1(C(=O)NCCN(C(=O)C(C)SC(F)(F)F)CCOC)[nH]ccc1C1CC1 CN=c1[nH]c(=NCc2nc(C3CCOCC3)cs2)[nH]c(=NCC(C)CCO)[nH]1 C1(NC(=O)CN2CCOCC2)CC2CC(NC(=O)C(Cl)=CCl)C2C1 c1(N2C(CCNC(c3cc(CC)n(C)n3)=O)CCC2)ccc(Br)cc1[N+](=O)[O-] c1(C(N2C(CNC(C3CCN(C)C3)=O)CN(C)CC2)=O)cnc2c(c1)nnn2C O=C1CCC2(C(=O)NCCCNC(=O)CCCn3ccccc3=O)CCCC2C1 c1(SCCC)cc([N+](=O)[O-])ccc1C.C1(C)CC(=O)ON1CC(=O)OC CCC(CC)(CCNC(C1CC(=O)N(c2nccs2)C1)=O)NC(C12CC(C1)C2)=O c1(CN2CC(n3cc(C(C)(C)N(C(CCC)=O)C4CC4)nn3)C2)cc(O)nc(O)n1 N1(CC=C)CCC(NC(=O)C(C)NC(c2cc(C)[nH]c2C)=O)CC1 c1(OC)ccc(C(N2CCC(CO)C(NC(=O)C(C)C)C2)=O)cc1F C1(CC)(NC(=O)CCc2ccn(C)n2)CCCN(C(C2CC2c2cnc[nH]2)=O)C1 C(=O)(NNc1nc(OC)nc(-c2ccccc2)n1)c1ccc(OC)c(OC2CC2)c1 N1(C(CC(=O)NCC)=O)CC(NC(=O)CC2CCCCC23CC3)C2CC2C1 c1(CN2C3C(C(N4CC(O)C4)=O)C(C3)C2)cc(Br)cc(Br)c1 N1(C(CCOCC#C)=O)CCC(NC(C2CC(O)(C#C)C2)=O)C(CC)C1 CC1CN(C(C2(c3cccc(F)c3)CC(N)C2)=O)CC2(CC2)C1 c1(OC)ccc(C(=O)NC2CCCC2n2cc(CCCCO)nn2)c(I)c1 c1(C(N2CC(C(=O)NC3CCN(c4ccccc4)C3)C2)=O)nccnc1OC N1(C(N)=O)CCN(C(c2cn(CCNC(c3cccc(O)n3)=O)nn2)=O)CC1 c1(NC(c2cncn2C(F)(F)F)=O)ccc(I)cn1 C1(NC(C2(C(=O)OCC)CCCC2)=O)CC(C)N(CC)C1.C12CC(F)(C1)C(=O)N2 C1(CNC(c2cc(C3CC3)on2)=O)CCC(NC(C2CCCC2)=O)C1 C1(C(N(C(CC)COC)C)=O)CC(O)CN1C(=O)C(C)CC c1(C(N(C2CCCN(C(c3c(C)nn(C)c3)=O)CC2)C)=O)ccc2cccnn12 C(=O)(C1=Cc2ccccc2C1O)NCC(C)N(C)C(c1conc1C(F)(F)F)=O N1(C(c2cc(OC)n[nH]2)=O)CCC2CCN(C(=O)CC(O)c3cc(C)cs3)C2C1 N1(C(COCC(=O)OC)=O)CCC(F)(CNC(=O)CC2CC(O)C2(C)C)CC1 CCC(C(=O)N1CC(CC(=O)NC(C)CO)C1)c1ccccc1 C1(C(N2CCOC(CN(C(=O)CCc3cc(Cl)cs3)C)C2)=O)(CC)CNC(=O)C1 CC(C)C(C)C(N)CNc1ccc(O)cc1 c1(C(=O)NCCNC(c2ccc3ccoc3c2)=O)nc2ncc(Br)cn2n1 c1(OC(C)C)cncc(C(=O)NCC2CN(C(C3CC3C#N)=O)C2)c1 Cc1ccc(C(N2CCN(C(c3cc(Br)cnc3Cl)=O)CC2CC#N)=O)c(O)c1 c1(NC(CC)CS(C)(=O)=O)cc(=NC2COc3ccccc3C2)[nH]c(COC)n1 C(=O)(C(F)C(F)(F)C(F)(F)F)N1CCC(CC(C)NC(c2c(C)snn2)=O)CC1 n1(C(CC)(C)C)nnnc1C(CC1CCCOC1)NCCCNC(=O)OC n1(CC)c(COC(C)C(=O)N2CC(Oc3ccc(Cl)cc3)C2)nc2ccccc12 C1(NC(c2cccnc2Br)=O)CC2CN(C(c3ccc(C4CC4)nc3)=O)CC2C1 C1(N(C(=O)C(C)C2CCCC2)CC#C)CCN(C(=O)C(F)=C2CCCC2)CC1 C1(C(=O)NCCCNC(=O)NC)CN(C(=O)C(O)CC(C)C)CC1C1CC1 C(C1CCCN1C(=O)C(F)=C1CCC1)=CC(=O)N(C(c1nn[nH]n1)C)C.C1C(C)C1 C1(NC(c2nnn(C(C)(C)C)n2)=O)CCN(C(=O)CCCc2ccsc2)CC1CO Cc1c(Cl)cnn1CC(=O)NCCNC(C1CCCN(C(=O)C(C)CN(C)C)C1)=O C(C(C(=O)NC(c1cnn(C)c1)C)C(C)C)NC(c1cc(CCC)on1)=O C12(C(=O)NCc3cn(C(C)C)nc3)CCC1CN(C(=O)Cc1cncnc1)C2 CC(C)CC(C(=O)NCC12CC(CN1C(C1(C3CCCO3)CC1)=O)C2)C(C)C Cn1nnc2c1CCN(C(C1(C)C=CCN1C(=O)C(O)C1CCCC1)=O)C2 C1(OC)CC(F)CN(C(=O)C(C(C)C)NC(=O)CC2OCCO2)C1 C1(C(=O)NCCN(C(=O)C=CSCC)CC)CC(Cc2ccco2)C(O)C1 c1(C(=O)NCC(CC)NC(c2c(C)noc2C)=O)c(F)cc(OC)cc1F N1(C(C(C)OC)=O)CCC2(C1)c1[nH]cnc1CCN2C(c1coc(O)n1)=O c1(SC(C(CC)O)C)cc(CN)cc(C(=O)NC(C)C)c1 Cc1ccccc1C(F)(F)C(=O)NC(C)C(C)NC(c1cnn(C2CC2)c1)=O C=CCC(C)(CC)C(=O)NCC1(NC(=O)CC(C=C)CCC)CCCCC1 C(=O)(CC(O)COC1CC1)NC1CC(CNC(c2cn(CC(C)C)nc2)=O)C1 c1(OC)ncc(F)c(=NC(=O)C2CC2C(=O)Nc2ncc(C(F)(F)F)c(Cl)n2)[nH]1 C(CC(CC)C(=O)NC1COCC1C(=O)N(C(C(N)=O)C1CC1)C)=CC C(=O)(CC(C)(C)C1CC1)NC1C(NC(C(CC)OC2CCCCC2)=O)CCC1 c1(NC(N2CCC(C(C(=O)NCCCC(=O)OC)C)C2)=O)c(C)cccc1C CN1C(=O)CCc2ccc(C(N3CCCC(C#N)C3)=O)cc21 Cc1cc2nc(NC(C)CCNC(=O)C(O)Cc3cnc[nH]3)cc(=O)n2o1 c1(NCCCC(CC)O)ncc(S(=O)(=O)NC2CCC(C)(C)C2)cc1Cl C1(NC(c2c(CC)nn[nH]2)=O)CC12CCN(C(=O)CC(C)c1ccco1)C2 c1(N(CCCNC(c2cc(C(C)(C)C)ccn2)=O)CC)ccnc(C#N)n1 C1(N(C(=O)C(CC)c2cccnc2)CC#C)CCN(C(=O)C(C)(C)CC)CC1 N1(C(c2scc(C)c2)=O)CCC(CNC(=O)CCC(=O)N2CCOCC2)C12CC2 c1(C(N2CCC(C)C(NC(c3ccc[nH]3)=O)C2)=O)cc2nnn(C)c2s1 c1(C(=O)NC2CC(C)(NC(CCC=C)=O)C2)ccc(Cl)c(S(C)(=O)=O)c1 C1(C2(C(N(CC(CN(C(C(c3ccnn3C)C)=O)C)O)C)=O)CC2)CCCCO1 C=CC1OCCC1C(=O)NC1(CO)CCN(C(=O)CCc2cnn(C)n2)C1 c1(C(N2CCCC(NC(CSCC=C)=O)C2C)=O)csc(S(C)(=O)=O)c1 C(=O)(C(CCF)NC(=O)CS(=O)(=O)NC)N(CC)Cc1ccoc1 N1(C(C2CCCSS2)=O)CCCCC1C1CCCN1c1ncc(I)cn1 c1(C(=O)NCC2C(CNC(c3ccc(OC)cc3)=O)C2)c[nH]c(=N)nc1C N1(c2c(Br)cnc(C(C)C)n2)CC2CCC(NC(c3ccns3)=O)CC2C1 C1(CC(=O)NCCC(C)NC(C2CCCC2F)=O)CCCC(=O)N1 C#CCCC(C(=O)NC1CC(C(N)=O)C1)NC(=O)C(C)C1(O)CCC1 c1(C(C)C(=O)Nc2ccc(OC3COC3)cc2)c[nH]c2ccccc12 C=C(Cl)CC(C(=O)Nc1cc(O)ccc1F)NC(c1cccnn1)=O N1(C(CC2CCC(=O)N2)=O)CCC2(CC(NC(=O)COC3CC3)C2)C1 c1(CCC(=O)NCCCCN(C(=O)COc2ccsc2)C)ccc(F)nc1 n1(C(C)C)ncc(Br)c1C(=O)NC1CC(NC(=O)C(C)(C)CO)CC1O c1(C(=O)OC(C)(C)C)cccnc1N1CCC(CC(=O)Nc2cc(C(N)=O)[nH]n2)C1 Cc1cc(NC2CCSC2)ncc1S(=O)(=O)NC(c1ccc2occc2c1)C Cc1occc(=O)c1OCC(=O)N(CC(O)CNC(C1CC1C(C)O)=O)C C(CC(O)C(=O)NC(C1CCN(C(C2CC23CCC3)=O)CC1)(C)C)SC CC1CC(NC(C2CCC(C)(C)C2)=O)CCN1c1ccc(C#N)nc1 C1(CNC(c2c(Br)cn(CC)n2)=O)CC(NC(C2CC(OC)C2)=O)CCO1 c1(N2CCC(CNC(c3cc(SC)on3)=O)C23CCC3)cccc(F)c1[N+](=O)[O-] CCC(C)C(C(=O)N1C(C(N)=O)CCC12CC2)N.N1(C(=O)C=CC(C)(C)C)CCCC1 C(CCCCCN(C(=O)Cn1nnnc1C(C)C)C)NC(c1c(C)scn1)=O C#Cc1ccc(C(=O)NC2CCN(C(c3c(Cl)ccc(C)c3N)=O)C2)cc1F N1(C(COCCC=C)=O)CC2(CCN(C(c3ccc(C(C)C)c(Cl)c3)=O)C2)C1 c1(OCCC)nc(C)ccc1C(N1CC(NC(C2CC2C2CCCO2)=O)C1)=O CC1(C(=O)NCC2CCN2C(=O)CC=C(Cl)Cl)COc2ccccc2O1 c1(CC(=O)NCCCC(C)NC(c2ncncc2Cl)=O)ccc2c(c1)CCC2 CON(C)C(=O)C1(NC(=O)C(C)(C2CCC2)NC(C2CC(C(C)C)C2)=O)CC1 C1(CNC(CCc2onc(CSC)n2)=O)CCN(c2ncncc2Br)CC1C c1(CC(N2CCCC(N(C(CCOC)=O)C)C2)=O)ccc(S(=O)CCOC)cc1 C1(NC(C(=O)Nc2ccc(SCC)cc2)=O)CCCC(C(C)C)CC1 C1(CC=C)(NC(=O)C(C)CNC(=O)CCc2cnoc2)CCCC1 C(=O)(C(C)(C)CCCNC(c1nnsc1N)=O)NCC(C(CC)CC)O c1(N(CCCNC(c2nc(C)oc2C)C)C)ccc([N+](=O)[O-])c(OC(C)(C)C)c1 N1(C(c2cc(COC)on2)=O)CCN(C(c2ccc([N+](=O)[O-])cc2)=O)C2CCC12 c1(C(N2CC(CC=C)(NC(=O)CC3CCCC3C)C2)=O)coc2c1COC2 C1(C(=O)NC2(C)CCN(C(c3c(C)n(CCO)cc3)=O)C2)Cc2nncn2C1 C(C)(C(CC(=O)NC1CC2(CCC2)C1O)NC(C1CC2CCC2C1)=O)OC c1(C(C)=O)cn(CC(=O)NCCCCCNC(C2CCCC2)=O)nn1 C1(CNC(CCC=C)=O)CCCCN(C(c2cc(CC)ccc2C)=O)CC1 c1(C(=O)OC)ccc2c(c1)CC(C)N2S(=O)(=O)c1c[nH]c(C(=O)O)c1C c1(OC)cc(C(=O)NC2(CNC(=O)C(c3cccc(Cl)c3)O)CC2)cnc1OC c1(C(N2CC(OCC(=O)NC(C)CCO)C2)=O)cnn(C)n1 C1(C(=O)OCC)OCCN(C(=O)C2CC2)CC1N(CC(=O)NC1CCCCC1)C c1(NC(C2(C)N(C(c3cc(C(C)C)on3)=O)CC2)=O)cc(F)c(Br)c(F)c1 CCC(CC)(C(N)=O)NC(C1(C)CCN(C(=O)CC2CC(C)=NO2)C1)=O C1(C)(C(C)C)CCN(C(=O)CCCCN(C(=O)C(C)(C)C(N)=O)C)CC1 C(=O)(CC(O)CC(C)(C)C)NC1CCC(CC(=O)NCCC#CCC)C1 c1(NC(c2ncc(C)s2)CC)nc2ccccc2nc1NCC1CCC(F)(F)C1 c1(C(=O)NCC2CC2CF)nc(C=O)cs1.C1(NC(C2(C#N)CC2)=O)CCOC1 N1(CC(=O)NCC2CC(C)(C)CN2C(C2CCCCS2)=O)C(=O)NC(C)(C)C1=O N1(C(C=C(C)C)=O)CCN(C(c2cc(C)cc(C)n2)=O)C2CCC12 N1(C(C(c2c(C)noc2C)(C)C)=O)CC(NC(C2CC2(C)Br)=O)CC2(CCC2)C1 c1(C(=O)NCC(O)CNC(=O)C(F)(F)C2CCCC2)cc2ccccc2[nH]1 c1(C(N2CC(N(C(CCOC(C)=O)=O)C)C2)=O)nc2sc(C)cn2c1C C1(CNC(CS(CC)=O)=O)CC2(CCN(C(C3CC34CCOCC4)=O)CC2)C1 C1(NC(=O)CCCC2CCC2)CCCC12CCN(C(c1ccoc1C1CC1)=O)C2 c1(C(=O)NCC(C)(C)NC(C(CC(=C)C)C)=O)cn2cccc(Br)c2n1 N1(C(C2N(C(CCC)=O)CSC2)=O)CCOC2(CCN(C(c3ccoc3)=O)C2)C1 O=C(C1=CCC(NC(c2cscc2Cl)=O)C1)NCc1ncccn1 N1(c2scc(CC(=O)OCC3(C)CC3)n2)CCCNC1=O.C(=O)C=CBr C=C(C)CN=C(NCc1cncnc1)N(C)CC(C(C)C)OC c1(C(=O)NC(C2CCCN(C(=O)Cc3cc[nH]n3)C2)C)cc(N(C)C)ccc1F C1(NC(c2c(C)nc[nH]2)=O)CCCC12CN(C(c1ccccc1CO)=O)C2 N=c1ncn(CC(=O)NC2CN(C(=O)CSc3cccnc3)C2)[nH]1 Cc1cc(C2(C(=O)NCC3CCN3C(=O)CCc3cnn(C)c3)CC2)on1 c1(C(N2CCC(C)CC2CNC(C2CCCS2)=O)=O)ccc(S(N)(=O)=O)c(Cl)c1 C12(OC)CCC(C(N3CC(O)CC3CNC(=O)Cc3ncccc3C)=O)(CC1)C2 N1(C(CC(C)OC)=O)CC2CC(NC(c3cncc(-c4ccccc4)c3)=O)C1C2 c1(C(=O)OC)cc(S(=O)(=O)NC(C(F)(F)F)c2ccc(C)o2)cs1 C1(CNC(=O)CC2CS(=O)(=O)C2)CC(O)CN1C(=O)CCc1cn[nH]c1 Cc1ncc(NC(=O)C(CCC2CCC2)NC(=O)CC2CC3CC3C2)c(C)n1 N1(C(C2C(C)OC(C)C2C)=O)CC2CC(C1)N(C(c1ccnnc1Cl)=O)C2 c1(COC)nc(CC2CC(CF)C2)n(-c2cccnc2OC)n1.C1(C)CCCC1 CC1CCC(CCCC(=O)NCC2(CCNC(=O)CC(F)F)CC2)C1(C)C c1(C(=O)NCCC(=O)NC2(C)C(C)C2)cc(C#N)cc2ccccc12 C(C)(CC1CCC1)(C(=O)NCC1CCN(C(=O)C(c2ccccc2)SC)C1)OC C1(CN)CC2CCC1N(Cc1nnc(-c3cc(O)c(Cl)cc3Br)o1)C2 c1(C(N2C(CCNC(C(CSC)(C)C)=O)COCC2)=O)cncc2c1CCCC2 C1(N(C(CC2(CN(C)C)CCC2)=O)CCO)CCCN(C(C2CC=CCC2)=O)CC1 c1(OCCOC)cccc(C(N2CCC(CC3CCCCN3CC(C)C)C2)=O)c1 c1(C(N(C2CCCN(C(=O)C3CC3)C2)CC)=O)ccc(Cl)c2c1OCCO2 N1(C(c2c(C)cc(F)s2)=O)CCC2(CC1)CCN(C(=O)Cc1cnco1)C2 Cc1ccnn1CC(N1CCCC1C(C)NC(C1(CN(C)C)CCCC1)=O)=O S(=O)(=O)(c1cccc(-c2ccccc2CO)c1)NCC1CNC(=O)O1 CC(CC(=O)c1ccc(F)cc1)C(=O)N1CC2(CCN2C(=O)C(O)CC2CC2)C1 N1(C(CCc2cc(C)n(C)n2)=O)CCN(C(=O)CCCCCO)C(C(C)C)C1 CC1CCC(NC(=O)Cn2ccc([N+](=O)[O-])n2)CN1C(=O)CC(C)C(F)F c1(C(N(c2ccnn2CC2CC2)C)=O)cc(C(=O)O)c(C2CC2)nn1 c1(CCC(=O)NCC(C2CC2)NC(CNC(CCC)=O)=O)c(C)noc1C C1(C(N(CC(C)NC(C2(CCF)CCOCC2)=O)C)=O)CCc2nnc(O)n2C1 C=CCC(C)(C)C(=O)NC1CCC1NC(c1ncc(C)cc1C)=O NS(=O)(=O)CCCC(=O)N1CC(C2(NC(C34CCC(OCCO)(CC3)C4)=O)CC2)C1 CC1CCN(C(=O)C(c2ccccc2F)C)CCN1C(c1cncc(Cl)c1)=O C=CC(CC)CC(=O)NC1CCN(C(=O)CSc2ccc(C(C)=O)cn2)C1(C)C N1(C(=O)Nc2n(C)cnc2-c2ccccc2)CCCC2CNC(=O)C12 C(CC(=O)N1CCC(C(N2CC3(C2)CN(C2CC2)C3)=O)O1)=CC Cn1ccc2cc(C(N3CCCC(CNC(=O)CCC(C)(C)F)C3)=O)cnc12 c1(C(N(CC(C)NC(c2cc(F)n[nH]2)=O)C)=O)ccc(C(F)(F)F)cn1 N1(C(C)=O)CCOC(C(=O)N(C)CC2CN(C(c3ccncc3O)=O)C2)C1 c1(C(=O)NCC(CCCC)NC(=O)C(CCC)NC(N)=O)ccn2ccnc2c1 c1(CC(=O)N(C)CC2(NC(C3CCCCO3)=O)CC2)cc2ccccc2c(O)n1 n1(CCC)ccc(C2c3nnnn3C3CC(C3)C(=O)N2)n1.C1(C)CCCOC1.OC C1(N(C(=O)C(O)CNC(=O)C=CC2CCCC2)C)CCCC1C#N CC1CCc2nc(Cl)nc(N3CCC3CNC(c3nccn3C)=O)c2C1 N1(C(C=C(C)CNC(=O)C2=CCCC2)=O)CCOC(C)(C)C1C n1(C(C)C)nncc1C(N1CC=CC1CNC(=O)C(C)NS(C)(=O)=O)=O N1(C(c2n[nH]c(CC)c2Br)=O)CC(NC(=O)C(C)CO)CC2(CCC2)C1 Cc1cc(OCC(=O)NCC=CCNC(=O)C=Cc2nnn(C)n2)ccc1[N+](=O)[O-] N1(C(CC2C(C)(C)C2)=O)CCC2(CCN(C(c3coc4c3CCCC4)=O)C2)C1 c1(C(N2CC(C)C2)=O)ccc2[nH]c(C(=O)NC(c3cnccn3)C)cc2c1 CC(C)C(C(=O)NCC(O)CNC(C1CCCC1C(F)F)=O)NC(N)=O C1(C(=O)NCCN(C(CCC2OCC(C(=O)OC)C2)=O)C)CCCCC1(C)C C1(C(=O)OC)OC2(C)CC1(CNCc1cc(C)cnc1O)C2 CCC(F)C(=O)NCC1C=CC(NC(C2CC(F)(F)C2)=O)C1 c1(CN2CCC(C#N)(NC(=O)CO)C2)ccc(O)c(F)c1F Cc1cc(C(=O)N(C2CCC(NC(c3nocc3C(C)(C)C)=O)C2)C)nc(O)c1 C(C1CN(C(=O)CN(C(=O)COC)C)CC1C(=O)NC1CC(Cl)(Cl)C1)=CC c1(N(CC(C(C)C)C)C)ncc(S(=O)(=O)NCC2(C)CSC2)cc1Cl C1(NC(C(C)SCCCC)=O)CC=C(C(=O)NCc2nc(C)sc2C)C1 N1(C(C2CN(CCOC)C(=O)C2)=O)CCCC(C2CN(C(c3cc[nH]n3)=O)C2)C1 c1(N(C)C)nc2ccc(C(=O)NC3COC4(C3)CN(C(=O)CC#N)C4)cc2o1 CCCCC(CNC(c1ccccc1Cl)CCO)CC C(C1=NOC2CCCCC12)N(c1ccccn1)C(=O)COc1cccc(F)c1 C12(NC(CSCC)=O)CCCCC1N(C(c1cc3cc[nH]c(=O)c3s1)=O)CC2 C1(C(N2CC(CC)C(O)C2)C(=O)NCCCCCC)CCOC(C)(C)C1 C(=O)(C1CCc2cccnc21)N1CCN(C)CC1CNC(c1cc(C#N)c[nH]1)=O CC(C)C(C#N)C(=O)NCCNC(c1coc(CSc2ccccc2Cl)c1)=O Cc1cncc(C(=O)NC2CCCC2NC(C2CC3(CCC3)C2)=O)c1 c1(C(N(C(CC)CNC(C2CC23CCC3)=O)C)=O)cc2cccnn2c1 N(C1CCc2c(Br)cc(F)cc21)C(C(CCSC)N)=O C(=O)(C1=CC2CCC1C2)NC1CC2CN(C(C3(C#N)CCC3)=O)C1C2 c1(CC(=O)NC(C2(O)CN(C(C3CC4CCC4C3)=O)C2)C)ccc(C(F)F)cc1 c1(C(=O)NC)cccc(C(=O)NC(CO)C(C)NC(c2ncoc2C)=O)c1 c1(C(=O)NCC(C2CC2)NC(C(C(C)O)N(C)C)=O)cnc2[nH]cnc2c1 c1(C(C)NC(C(=O)Nc2cn(CC=C)nc2)=O)cccc(N2CCCC2=O)c1 C(=O)(C1=CCc2ccccc21)NC1C(C)CN(C(=O)COCCCN=[N+]=[N-])CC1 c1(OC(C2C(CNC(COCCC=C)=O)C2)=O)cc(CC)on1 Cc1cc(NC2CCC(N(C)C(C3CCCC(C)CC3)=O)CC2)n2ncnc2n1 C#Cc1cncc(C(=O)NCc2cc(O)cc(F)c2)c1.C12(CCCC1C)C(=O)N2 N1(C(CC(CCC)CC)=O)CC(C2CCCN(C(C3CC3C(C)O)=O)C2)C1 C12(C(=O)NC3CCC(C(C)C)CC3)CCCC1CCN2C(c1cnn(C)c1)=O C1(C(=O)NC(C2(O)CCCCC2)C(=O)NCC(COCC)O)CC(=O)CC12CCC2 c1(CC(=O)NC2CC(CCNC(C(C)SCCC=C)=O)C2)ccnc(O)c1 c1(C(CNC(=O)C=C(Cl)Cl)NC(C2CC(F)(F)C2)=O)ccc(F)cc1F C(CC(CC)C(=O)N(C)CCNCc1c(C(=O)N(C)C)ccs1)=CC c1(C(N2CCC(NC(c3cc(Br)c[nH]3)=O)C(F)C2)=O)cc(Br)cc2ccccc12 N1(C(C(=O)NC(c2cc(C)cc(C)c2)C)=O)CC2CCN(C)CC(C2)C1 C(=O)(CCC(CF)CF)N(C1CCN(C(=O)C(C)C(C)(F)F)C1)CCC C=C=CC(C)C(=O)NCCC(CNC(c1cc[nH]c1C)=O)OC C1(CNC(C(C)O)=O)CN(C(c2cc3scc(Br)c3[nH]2)=O)CC(C)(C)O1 C1(c2n(CC)c(O)nn2)CCCN1N1CC(C)(C)OC2(CCC2)C1 c1(C(N(CC(C)NC(=O)CC(C)(C)C#N)C)=O)ncn2cc(Cl)ccc12 C=CCC(C)C(=O)Nc1ccc(Oc2cnccn2)cc1 C(CN=c1cc(C)nc(NC(C)Cc2ncn(C)n2)[nH]1)SCC C1(C)(C(=O)NCCCN(C(C2C(C=C)C2)=O)C(C)C)CCNC1=O C(N=c1cc(NCC(C)(F)C(C)(C)F)nc[nH]1)c1[nH]nc(C(C)C)n1 c1(OCC)cc(C(N2CCCC2CNC(C2CC2c2ccccn2)=O)=O)ccn1 C1(NC(CC(C)SC)=O)CN(C(=O)CNC(=O)CC(F)(F)F)C2(CCC2)C1 N1(C(c2nc(COC)sc2)=O)CCOCC1CNC(=O)CCc1cccs1 c1(OCC)cc(NC(c2csc(NC(=O)CCc3ccc(F)nc3)n2)=O)ccn1 C12(NC(CCN(C)CCO)=O)CCOCC1CN(C(=O)Cc1cn(C)nn1)C2 c1(C(N(CCCCCNC(C2CC23CCC3)=O)C)=O)n[nH]c2c1CC1CC21 C1(NC(C(c2c(F)cccc2F)C)=O)CCCCN(C(=O)CSCC(F)(F)F)C1 C1(NC(Cc2ccc(C)cc2)=O)CCCCN(C(=O)C(=O)NCC(F)F)C1 c1(N(CCNC(=O)OC(C)(C)C)C(C2CCOC2)=O)cncc(Br)c1 C1(CN(C)C(c2cncn2C2CC2)=O)CCCC2(CC2)C1 c1(C(=O)NCC(CC=C)NC(C2(C3CC3)CCC2)=O)c(C)ncn(C)c1=O C(CCCC(=O)N(C)CC1CCCN1C(C1(C)CS(=O)(=O)C1)=O)SC Cc1cn2cc(C(=O)NCC(O)CNC(=O)C(C)S(C)(=O)=O)ccc2n1 C(=O)(C(C(=O)N(CC(C)NC(=O)C(F)(F)c1cscn1)C)C(C)(C)C)OCC N1(C(CS(=O)(=O)NCC)=O)CCC(NC(=O)CCCCCN(C)C)C12CC2 C1(CNC(C(CNC(C(c2cnn(C)c2)C)=O)(C)C)=O)CCOCC1(C)C CCC(CCCC(=O)NCC(C)(O)C1CC1)NC(c1cnc(OC)cn1)=O Cc1ncnc(C)c1CC(=O)NC1CC12CC(NC(=O)C=CC(C)C)C2 Cc1ccc(F)c(C(=O)NCC(c2cn(C)nn2)=O)c1 Cc1nc(C)c(C(=O)NCCC(C)CCNC(=O)Cc2cncc(Br)c2)o1 c1(C(C)(C)C)cc2c(Nc3ccccc3C(=O)NCC3CNC3)ncnc2s1 c1(C(=O)NCC(C)CNC(c2cnn(C3CCC3)c2)=O)c(Cl)ccc(Cl)c1O C1(C(C)NC(c2ccccc2)CO)C(C)(C)C1(C)C c1(C(=O)NC(C)(C)CNC(=O)C=Cc2ccc[nH]2)cnc(O)c2cnccc12 C1(N(C(=O)C(C)N2CC(C)C2)CC)CCCN(C(=O)CCn2cccn2)C1 C1(NC(C(CC)F)=O)CC2(CCN(C(=O)CCN3C(=O)CCC3=O)CC2)C1 Cn1ncc2ccnc(C(N3CCN(C(C4CCC(=O)O4)=O)CC3CCO)=O)c12 c1(C(=O)NC(CNC(C=C(COC)C)=O)C2CCC2)cnc2ccccn2c1=O O=C(C#CC1CCCCC1)N1CC2CC1CN2C(c1c(Cl)ccc(O)c1Cl)=O CCC(C)C(=O)N(CCOCC)CC.C12(C)CC(C1)NC2=O.C(C)(=O)O C1(C(=O)NCC2C=CC(NC(CCC=C=C)=O)C2)CCC(=O)N(CCOC)C1 N1(C(C(C(C)O)N(C)C)=O)CCC(C2CN(C(c3ccc(=O)n(C)n3)=O)C2)CC1 c1(OC)cncc(C(N2CCC(C3CCCCN3C(c3cc(CO)on3)=O)C2)=O)c1 C1(C)(COC)CC(NC(C2CC(C)(C)C2)=O)CN1C(c1c[nH]cc1Br)=O c1(C(N2C(CNC(Cn3cc(C(=O)NC)nn3)=O)CCC2)=O)cc(C)n(C)n1 c1(OC)cc(C(=O)NC2CN(C(C3CC(C(F)(F)F)C3)=O)CCC2F)ccc1O c1(C(N2CC(C(C(N3C(C(=O)OC)CC3C)=O)O)C2)=O)ccc(Br)cc1 c1(C(=O)OC)ccc(C(F)(F)F)nc1N(C1CCCCC1c1ccccc1)C CCC(C(=O)N1CCC(C)CC1CNC(c1nnn(C)c1N)=O)C(C)(C)CC CCC(C)CCCC(=O)NC1CCCCC1NC(c1cn(CCOC)nc1C)=O c1(C(=O)NC2C(NC(=O)CCC3CCOCC3)CCC2)ccc(O)c(F)c1F CCCC(C#N)C(=O)NCC(C)(C1CC1)NC(=O)COc1cn[nH]c1 c1(C(N2CCN(C(C(CC)OC)=O)CC2CC)=O)nn(C)cc1[N+](=O)[O-] c1(OCC)cc(Br)cc(C(N2CCCCC(NC(C3(C)CC3)=O)C2)=O)c1N C12(NC(c3ccc(CCC)cc3)=O)CCCN(C(=O)CO)CC1C2 C1(CNC(C(c2nc(C)sc2)=O)=O)(NC(C2CCC2)=O)CCC(C)(C)CC1 O=C(CCCC1CC1)NCC1CCC1NC(c1ccnn1C(F)F)=O c1(C(N2CCN(C(C3(CC)CC3)=O)CC2CC(F)F)=O)ccc2c(c1)C(C)CO2 N1(C(c2c(C)c(Cl)ccc2)=O)CCC(C2CC(NC(=O)C(F)C(C)(F)F)C2)CC1 C=CCC(C)(C)CC(=O)N(C1CCN(C(=O)CCC(C)(F)F)C1)CC c1(C(=O)NCCC2N(C(C(c3cnn(C)c3)C)=O)CCC2)ccnc(F)c1F N1(c2ccnc(NCc3c(C)ccc(F)c3)n2)C2CCC1CN(C)C2 c1(C(=O)NC(c2ccnc(C)n2)C)ccc(F)c2ncccc12 c1(CC(N2C(CC(=O)NC3CCC(F)(F)C3)COCC2)=O)c(F)cccc1F N1(C(c2c(COC)cc[nH]2)=O)CCC(C)(C)C1C(N1CC(COC(C)=O)C1)=O n1(C(C)C)ccc2cc(C(=O)NCCNC(=O)CC(O)C(Cl)(Cl)Cl)ccc12 Cc1cc(CN2CCCC2CNC(c2[nH]cnc2-c2cccnc2)=O)cnc1Cl Cn1cnc(C(N2CCC23CN(C(C2CCC4(CC4)C2)=O)C3)=O)cc1=O C1(NC(c2c(CC)cco2)=O)CC(NC(=O)CC2NC(=O)NC2=O)CC1O C#CC(C)(C)C(=O)N1CCC(C2OCCC2NC(=O)COCCOCC)CC1 c1(C(N2C(C(=O)Nc3ccc(Cl)cc3)CC2)=O)cc2cnccc2[nH]1 c1(C(=O)NC(C)C(C)F)ccn(CCNC(=O)CC(C2CC2)C2CC2)c1 C=Cn1nccc1C(=O)NCC(C)(C)CNC(=O)CNC(=O)C(F)(F)F c1(CNC(C2CCCN(C(COCP(C)(C)=O)=O)C2)=O)[nH]c2ccccc2c1Cl c1(OC)cccc(NC(c2cnc(-c3sccc3OC3CC3)cn2)=O)n1 c1(NCc2ccc(CC)o2)ncccc1S(=O)(=O)N1CC2CCN(C)C2C1 c1(OC)cnnc(C(=O)NC2COCC2CNC(=O)C(=C2CCCCC2)F)c1 CC1CN(C(C2(O)CCC2)=O)CC2(CCN(C(=O)CCCCCCN=[N+]=[N-])C2)O1 Cc1cc(F)ccc1C(=O)NC1C2CC1N(C(=O)C(F)(F)C(O)C1CC1)C2 c1(C(N2CCC(O)(CNC(c3c(C)occ3)=O)C2)=O)cc(C(F)(F)F)ncc1N CP(C)(=O)c1cccc(CNC(N2CC=CC2Cc2ccc(Cl)cc2)=O)c1 C12CN(C)CCCN1C(=O)C(OC)CCSCC2C.C(=O)(C(=O)C(C)(C)CC)OC N1(C(c2c(C)cncn2)=O)CCC2(CC1)CC(C)N(C(C1CC1(Cl)Cl)=O)C2 c1(CSCC2CC(CNC(C(C)C(=O)CN3CCCC3COC)=O)C2)ccccc1 C(c1ccc[nH]1)=CC(=O)NC(C1CCN(C(c2ccc(N3CCC3)s2)=O)C1)(C)C c1(C(=O)NC(C(C)C)CNC(=O)C(C)CC2CC2)ccc2c(n1)NCC(=O)N2 N1(C(COCCCC(C)C)=O)CCCC2(CCCN2C(C2CSCCS2)=O)C1 c1(C(N2CC3C(CNC(CCC=C=C)=O)(C3)C2)=O)ccc(N)cc1Cl C1(CNC(c2c[n+]([O-])ccc2O)=O)CCCCN(C(=O)Cc2nc[nH]n2)C1 N1(C(c2nc(C)n(C)n2)=O)CC2CC(CNC(=O)C(C)(C)c3cccs3)C2C1 Cc1nccnc1C(=O)NC(C)C(C)NC(c1cnccc1Cl)=O c1(C(=O)NC(CN(C(C2CC(C(F)(F)F)C2)=O)CC)C)cc(C)c(C)cc1N C1(C(=O)NCCOCCCNC(=O)C(=C2CCOCC2)F)C2CC3C(C2)C13 C1(NC(C(C)S(C)(=O)=O)=O)CN(C(=O)C2=CCCOC2)CC12CCOCC2 C(=O)(CCCC(N)=O)NC(C(C)NC(CCC(C)N(C)C)=O)C N(C(=NCCC1OCCC1C)NCc1cc(C(F)F)nn1C)CC(=C)C N1(C2CN(C(C(C#N)C3CC3)=O)C2)CC(NC(C2(O)CCC2)=O)CC1=O c1(C(=O)NCCCN(C(C2CCC(CO)CC2)=O)CC)cnn2ccc(O)nc12 c1(C(=O)NC(C)(CNC(=O)CCC2CC2(F)F)CO)ccc2c(n1)CCCC2 CC1CC(CNC)CN1C(=O)Nc1nccnc1-n1ccnc1 Cc1cc(C(=O)NC2CN(C(c3ccccc3F)C)CC2(C)C)c(F)cc1F C#CC(C(C)OC)NC(=O)CC(C1CC1)NC(c1ocnc1C(C)C)=O C1(C)(CC(=O)NCC(COCC)O)CCN(C(c2c[nH]nc2C)=O)C1 c1(NC(C(CNC(C2C(=C)C2)=O)(C)C)=O)ccc(F)cc1C CCCC(C)CC(=O)N1CCOC(C(=O)NCC2CNC(=O)CO2)CC1 N1(C(C(C(C)NC(C(C)C2CCC2)=O)(C)C)=O)CCC2(C=CCO2)CC1 C(C(=O)NC1(CNC(=O)Cc2ccsc2)CCC1)(C(C)(C)C)OCC(C)C N1(C(C2CN(C(=O)NC)C2)=O)CCC2(CCC2NC(=O)CSc2cn[nH]c2)CC1 c1(C(=O)NCCC(=O)NC(c2n(CC)ncn2)C)cccc(C)c1O C#Cc1cncc(C(Cc2ccccc2Cl)Nc2ccc(F)cc2C)c1 C(=O)(C(=O)C(C)CC)NCc1cc(C(N(C2CCC(=O)NC2)CC)=O)n(C)n1 C1(CNC(C2(C)CC3CC3C2)=O)CCCCN(C(C2(C#N)CCOCC2)=O)C1 Cc1ccc2[nH]cc(C(=O)N(C)CC3CCN(C(=O)CCc4cn[nH]c4)C3)c2c1 C1(NC(C(C(C)C)C2CCC2)=O)COC2CN(C(=O)C=CCN(C)CCO)CC12 C1(C(C)NC(=O)Cn2cnc(C(F)(F)F)n2)CCN(C(=O)C(C)(C)F)CC1 C1(C(N2CCC(CC(=O)NC3CC(C#C)C3)C2)=O)CC2(C1)CC(C)C2 N1(C(c2cc(C)oc2)=O)CCN(C(=O)CCC(C)(F)F)CC(O)C1 C1(COC)CN(C(=O)CC2(COC)CC2)CCN1C(c1cc(O)nn1C)=O C(C(C)CN(C(=O)C(C)N(C(=O)CC1CC=CC1)C1CC1)C)OC N1(C(CSC(=N)N)=O)CCC2(CC1)COC(CNC(c1nccc(Br)c1Cl)=O)C2 c1(C(=O)NC(C2CCN(C(C3CCCCNC3=O)=O)C2)C)cc(F)c(F)cc1N N1(C(C(C2CC(NC(c3c(COC)cc[nH]3)=O)C2)F)=O)CC(C)c2ccccc21 C#CC1(C(=O)NCCC(C)(C)CNC(c2cscc2CC)=O)CCCC1 c1(CN2CC(CN(C)C)C3(C2)CC3)cc(F)c(F)c(Cl)c1F N1(C(COc2c(C)ccc(CO)c2)=O)CCCC2(CCN(C(=O)C(C)(C)O)C2)C1 C12(C(=O)OCc3onc(COCC)n3)CCOC1CC(=O)NC2 c1(C(=O)NC2CN(C(C3C(=C)C3)=O)CC2(C)C)cc2c(cc1Cl)OCO2 Cc1nc(C(=O)NCC2CCN2C(=O)C(c2c(F)cccc2F)C)ccc1C#N C(=O)(C(C(C)C)NC(N)=O)N(C1CCN(C(=O)Cc2nc(=N)[nH][nH]2)C1)CC Cc1cc(N)ccc1C(=O)NC(CNC(c1csc(C)c1C1CC1)=O)C(C)C N1(C(CC2(COC)CC2)=O)CC2CC1CN(C(C13CCC(CC1)C3)=O)C2 Cc1nc(N(C)Cc2cn(C)nc2-c2ccccc2Br)c(Br)nc1Br C(CN(C)C)(C(=O)NCC(c1cc[nH]n1)O)NC(C1CC(OC)C1)=O C(CC(C)(C)CNC(=O)CN1C(=O)CCC1=O)NC(C1CC(SC)C1)=O c1(N2CCN(CC=C)C(=O)C2)nc(=N)[nH]c(=NC2COCC2CO)[nH]1 C#Cc1cnc(C(=O)NCCC2COCCN2C(=O)CC(CC)SC)c(C)c1 C1(C)(CNC(C(C2CCN(C(c3cc(C)no3)=O)CC2)C)=O)CC2(CCC2)C1 C1(NC(c2c(C)nn(CC)c2C)=O)CN(C(C2(C)CCOCC2)=O)CC2(CC2)C1 C1(CCCC)(C(=O)NCCOC(C)(C)CNC(=O)CC2CCSCC2)CCCC1 C1(OC)CC(CC(=O)N(C(CNC(C23CC(CCO2)C3)=O)C2CC2)C)C1(C)C N1(C(C(=O)NC(CN(C(c2c(C)c(O)ccc2)=O)C)C)C)CCc2ccccc21 Cc1nccc(C(N2CCC3CC23C(=O)NC(C)CCCCO)=O)c1C C1(C(N(CCCC=C)CC)=O)CNC(=O)CN1C(c1cc(COC)on1)=O c1(-c2c(C(N3CCN(C(C)=O)CC3C)=O)coc2)csc2c(O)ccnc12 C1(NC(c2cn(CC)nc2C2CC2)=O)CN(C(=O)COCCF)CCC12CCC2 c1(CC)cc(C(=O)NCC(=O)N(CC(=O)NOCC(C)(C)C)C(C)C)nn1C C(=O)(CCN(OC)C(=O)c1cccc(NC(c2ccccc2C)=O)n1)OC S(=O)(=O)(c1cc(Br)ccc1Cl)NCCCNc1c([N+](=O)[O-])cn(CC)n1 c1(C(=O)NC(CC)CNC(=O)CC2CC(F)C2)cc(O)nc2cnccc12 c1(C(=O)OC)cc(Cl)ncc1N.C12CC13CCN(C3)C2=O.c1(CO)ccc(CBr)cc1 C1(CNC(C2(COC)CC=CC2)=O)CCN(C(=O)C2=NOC(C)C2C)CC1(F)F N1(CC(=O)NCc2nc(C(=O)O)n[nH]2)CCC(N2CCCC2O)CC1 Cc1onc(C(N2CC3(CCC3)CC2CNC(=O)C(O)C(F)F)=O)c1[N+](=O)[O-] C1(C(=O)NC2CN(C(C(F)=CCC)=O)CC23CC3)COc2ccc(OC)cc2C1 C(=O)(CCCCNC(=O)C(=O)NC1CC1)NC(C#C)(C)C c1(C(=O)NCC2CC3CC3N2C(C2CCCCC2)=O)cc2c(F)cccc2[nH]1 c1(CC(C)C)ccc(C(=O)N(CCCCCNC(=O)C(F)C2CCOC2)C)s1 O=C(NNc1ccc(F)c(F)c1)C1CC(n2cc(C3CC3)nn2)C1 c1(C(N2CCCCC(NC(C3(COC)CCOC3)=O)C2)=O)cc(N)c(Cl)c(O)c1 Cc1cn2[nH]c(=NC3CCN(S(=O)(=O)c4ccc(Cl)c(Cl)c4)C3)ccc2n1 C1(C(=O)OC)(C(N2CCCC(C3CCCN3)C2)=O)CC2(CC(F)C2)C1 n1(CCC(=O)NCC2(NC(C3C4(CC4)C34CC4)=O)CCOC2)cccnc1=O c1(CNC(=O)COCC(F)F)ncccc1C(N1CCCC(c2ncc[nH]2)C1)=O N1(C(C(C=C)O)=O)CCC(C2CCC2)(CNC(c2cc(CC)ccc2O)=O)CC1 Cc1ccc(F)cc1C(N1CCC(C(=O)NCc2ccc(CO)cc2)C(O)C1)=O c1(OC)cc(C(=O)NCC(C)(C)CN(C)C(C2(C)CCCN2C)=O)cc(F)c1F N1(C(CN(c2c(CC)cccc2)C)=O)CCCC(CO)C1C=O C(CC)(C(=O)N=c1cc(-c2cccc(Cl)c2F)[nH][nH]1)NCc1cccc(CC)c1 CC1(C)C=C(C(=O)N2CCC(NC(C3C(F)(F)C34CCC4)=O)C2(C)C)C1 c1(C(=O)NC2CCN(C(C3(OC)CC3)=O)CC2C)ccc(C)c2ccccc12 c1(C(=O)NCCN(C(C2CN(C(C)=O)C2)=O)C)nnc2ccccc2n1 CCC(=O)CCC(=O)NCC1CCCC(NC(c2cc(C)n(CC)c2C)=O)C1 Cc1cc(C)c(C(N2CCCC(NC(=O)CCc3scnc3C)C2)=O)c(Cl)n1 c1(C(=O)NCC=CCNC(C2CCC2(F)F)=O)cc(Cn2cc(Cl)cn2)cs1 c1(OCC(C)C)ccccc1C(=O)NC1CC(CNC(=O)CCSC(F)(F)F)C1 N1(C(CC(=O)OCC)=O)CC2(CCC(NC(c3cn(C)nc3O)=O)CC2)C1 C12(CNC(CCS(C)(=O)=O)=O)CCCC1N(C(c1cc3ccccc3[nH]1)=O)CC2 N1(C(CC2ON=C(C)C2)=O)CC2(CO)CC1(C(N1CC(C(C)C)CCC1C)=O)C2 CC(C(=O)N(C)CCOCCC(N1CC(O)C(C)(C)C1)=O)S(N)(=O)=O CS(C)(=O)=Nc1cccc(C(=O)NCC2CCCCN2C(C2CC23CCC3)=O)c1 C1(C(=O)NC(C(=O)NCCCNC(=O)NC)Cc2ccoc2)CC2CCCC2C1 C1(CC(=O)N(C2CC(NC(C3(C(C)C)COC3)=O)C2)C)CCOC1(C)C C1(NC(C2(O)CCCC2)=O)CC2CN(C(=O)Cc3ccc(F)c(F)c3)CC12 n1(CC(=O)NCCN(C(CCN(CCC)C)=O)CC(C)O)nnc(C(C)(C)C)n1 C(C(CC(C)C)C(=O)NC1CCC(N(C)C(c2cnoc2C)=O)CC1)OC C1(C)(C(N(C2C(C)CCC2)CCCCCO)=O)CC2(CCOCC2)C1 c1(C(c2ccccc2)NC(c2csc(-c3cccs3)n2)=O)ccc(Cl)cc1 c1(NC2CC(CNC(C(C)=CC)=O)C2)ccc([N+](=O)[O-])cc1NC N1(C(CCCNC(=O)OC)=O)CCCC(CO)(NC(=O)CCC2(C)N=N2)C1 C1(C(N(CCCNC(c2c(SCC)cncc2)=O)C)=O)CC2(CCOCC2)C1 C1(C2CCN(C(c3ccncn3)=O)C2)(NC(c2sccc2Cl)=O)CC1 c1(C(=O)NCCN(C(C)C(=O)NCc2ccccc2)C)c(C#N)cnn1C c1(NC(c2ncccc2-c2cnn3ccccc23)=O)cccc([N+](=O)[O-])c1Cl CCC(CCOC)C(=O)NCc1csc(CNC(=O)C(c2ccc(Cl)cc2)O)n1 C(C(C)(C(=O)NCCC(=O)NO)NC(=O)CNC(=O)CN(C)C)SC c1(OC)ccc(NC(C2CC23CCN(C(=O)C=Cc2cnn(C)c2)C3)=O)cc1C CCC(C)C(O)C(C)C(=O)N1CCN(C(c2ccn(C)c2C)=O)CC(O)C1 c1(C(N2CCCCC(CNC(C(C)CF)=O)C2)=O)cncc2c1CCCC2 Nc1ccc(-c2ccc(CN3CCC(c4cc[n+]([O-])cc4)C3)s2)nc1 N12CCN(CC1)CCCSCc1cc(no1)C2=O.c1(C(=O)SCC)n[nH]cc1C c1(C(=O)NCC2C(C)CN(C(c3ccnn(C)c3=O)=O)C2)cccc2[nH]ccc12 C(C(CC(F)(F)F)NC(=O)CCC(N)=O)NC(COCc1n(C)ccn1)=O C1(NC(N)=O)CCC2(CCCN(C(=O)Cc3csc(=N)[nH]3)C2)C1.C12(CC1)C(=O)N2 CC1(C)COc2c(NC(=O)NC3(C)CCCCC3)cccc21 C1(CCC(=O)NCCCN(C(=O)Cn2cnnn2)C(C)C)CCCOC1 C1(C(=O)NC2(CNC(=O)CC3(N4CCCC4)CC3)CC2)CCOCC12CCCC2 Cc1nc2ccc(C(=O)NC3CS(=O)(=O)CC3C)cc2[nH]1 c1(C(N2CC(CC=C)(NC(=O)CC3CCCCCC3)C2)=O)cccc2c1OCO2 c1(C(=O)NC2C(CC)C2)cccc2c1OCCN2 CC1CCCCC1NC(c1cccc(Br)n1)CF Cc1ccc(C(N2CCCC3(NC(c4ccnnc4C)=O)CC3C2)=O)c(O)c1C C(CC(=O)NCc1cnc(C)[nH]1)(C(C)C)NC(C1(C(C)=O)CC1)=O CC(C)CC(C)C(=O)N1CCC(CNC(c2cnc(C3CCC3)o2)=O)CC1 C(=O)(C1=C(NC(C2CN(Cc3c(F)ccc(F)c3F)CCS2)=O)CCC1)OCC c1(COC(=O)NC(C(=O)NCC(CCOC)OC)(C)C)cnc(C)nc1 N1(C(c2ccc(OC(C)C)cn2)=O)CC(C)CN(C(=O)CSC2CCC2)C(C)C1 C1(C(N(CC(N)=O)CC)=O)CCN(C(C2(F)CCOC2)=O)CC1O C(CCOCCO)(C(=O)NC(c1cncs1)C)NC(CCC)=O C12(NC(C3C(C)C3C)=O)CCCCCC1N(C(=O)CCc1ccccc1Cl)CC2 c1(C(=O)NC(CNC(C(=O)NCC)=O)C(C)C)ccc(C(C)C)c(F)c1 C1(C2CCN(C(C3(CF)CC3(F)F)=O)CC2)(NC(c2ccns2)=O)CCC1 c1(SCC(N2CCC(C(C)NC(C(C)OCCCC)=O)C2)=O)nc(C)cc(C)n1 C(CCC1CC1)(C(=O)NCCCC(F)F)NC(C1C=C(C)CS1)=O c1(C(N2CCC(NC(=O)C(F)OC(F)(F)F)C(O)C2)=O)nccc2c[nH]nc12 c1(NC(c2nnnn2C(C)(C)CC)C2CC(=C)C2)cnc(C(C)C)nc1 N1(C(C(C)OC)=O)CCN(C(=O)Cc2c(C)nn(CC(C)C)c2C)C(CO)C1.CO c1(C(N2CCC(C(C)CNC(C3OCCCO3)=O)CC2)=O)cc2occc2n1C CN1CCCCC(C(=O)NC2CCC(NC(C3CC(O)CN3C)=O)C2)C1=O C12(C(=O)NC3(C)CC(F)C3)CCC(NC(=O)CC3CCSC3)(CC1)C2 N1(C(c2cn(CC)nn2)=O)CCOC2(C1)CN(C(C1CCCC13OCCO3)=O)C2 N1(C(C2N(C(C(CC#C)C3CC3)=O)CC=CC2)=O)CC2(CC2)CC1C#C C1(NC(C(CC)COC)=O)CC2CCC1CN(C(=O)C=CSc1ccccc1)C2 N1(C(C2C(C)C2)=O)CCC2C(CCN2Cc2ccc(F)c(Br)c2F)C1 c1(C(N2CC(NC(CS(N)(=O)=O)=O)C(O)C2)=O)cccc2[nH]nc(O)c12 N1(C(CCC(C)(C)O)=O)CC2CCN(C(c3noc4c3COCC4)=O)CCC2C1 c1(C(=O)NCC2OCC(CNC(CP(C)(C)=O)=O)C2)c(Cl)nc2ccccn12 c1(CC(=O)NC(COC(C)C)C(=O)NC2CCN(C(C)C)C2)ccc(O)nc1 C1(NC(Cc2c(C)ocn2)=O)CCCC(NC(c2cc(=O)n(C)o2)=O)CC1 c1(OC(C)C)ccc(C(=O)NCC2(O)CN(C(=O)CC3CC34CC4)C2)cn1 N1(C(C(CC#C)CC#C)=O)CC2CCN(C(c3oc(C)cc3Br)=O)CC2C1 c1(C(N(C)CC2C(NC(c3c(C)nn[nH]3)=O)CCC2)=O)onc2ccccc12 N1(C(C2(NC(N)=O)CC2)=O)CC(O)(c2cn(CC3(F)CCOC3)nn2)C1 C(CCCCC(=O)NCCc1cnn(C)c1C)NC(CC(CC)SC)=O Cc1cc(NCC(c2nnnn2C2CCCCCC2)NC(C)(C)C)cc(C)n1 C(c1ccccc1)=CC(=O)NC(CN(C(c1ncn(C(C)C)n1)=O)C)C C1(C(=O)NCC(C)(CO)NC(c2cc(F)c[nH]2)=O)CCC(c2ccccc2)CC1 C(=O)(C1=CSCCO1)NCCC1CC(NC(Cc2n[nH]c(=NC)s2)=O)C1 c1(CC(=O)NC2CCCC(CNC(C3(COC)CC3)=O)C2)ccc(O)cc1F N1(C(C2N(C(C(C)n3cnnn3)=O)CCC2)=O)CCC(C)(C)C(CO)C1 c1(OC)ccnc(C(=O)NCC=CCNC(=O)CC(C)(C)O)c1 N1(CCC(C)(C)C)CCC(CNC(=O)C(C)(O)Cc2ccccc2)C(C)(C)C1 O=C(NNC(=O)c1ccc(O)nn1)NCC1CCCN(CC(F)F)C1 CC1CC(CNC(=O)CC2CC2)CN(C(=O)C(C2(O)CCCCC2)(F)F)C1 N1(CC(=O)NCC2CC(C(F)(F)F)CN2C(c2cc(Cl)ns2)=O)C(=O)CNC1=O c1(CC(N2CCC(OC(C3(C#N)C(C)C3)=O)CC2)=O)ccc(OC2CC2)cc1 N1(C(c2c(C)nn(C)c2Cl)=O)CCN(C(=O)C(=Cc2c[nH]cn2)F)CC2(CC2)C1 C12(NC(C=CCOC)=O)CC1CN(C(=O)CC1C=CCCC1)C2 N1(C(c2cn(C)nc2C2CCC2)=O)CCC2CCCC(C1)N2C(C1C=CCC1)=O C(C(F)(F)F)=CC(=O)NCCC1(NC(c2cnn[nH]2)=O)CC1 Cc1ccc(F)c(-c2cncc(C(=O)NCCOC3CCCCC3)n2)c1O c1(-c2c(C)occ2)nc(C2CC(C)(C)C2)n(CCOCC(F)(F)F)n1 c1(C(N(C(=O)C(C2CCCO2)C2CCC2)C)=O)cccc(CCN=[N+]=[N-])c1 C1(NC(c2ccc(CC)c(Cl)c2)=O)CCC(O)CN(C(C2(N(C)C)CC2)=O)C1 C1(n2cc(CSCC(=O)Nc3ncc(Br)s3)nn2)CCCCC1C(=O)O c1(C(=O)NCC(C(C)C)(C)NC(C2CC(C)(F)C2)=O)cn(C)c(=O)n(C)c1=O c1(CCC(N2C(CC(=O)N(CC(O)CO)C(C)C)CC2)=O)cn(C)nn1 C12(CC(=O)N(C)Cc3cccc(F)c3)CCC1CN(C(=O)CC1(O)CCC1)C2 C(=O)(NNc1nc(Cl)ccc1Br)C1N(S(C)(=N)=O)CCC1 c1(C(=O)NCC2CC2CNC(=O)C(O)C(F)(F)F)cnc2c(c1)CCCO2 C(=O)(C1CCC(=O)c2cccn21)N(CCCC(=O)Nc1nc2ccccc2s1)C c1(C(N2CC(COC)(CNC(c3cc(C)c[nH]3)=O)C2)=O)cc([N+](=O)[O-])n[nH]1 C(CCC(C)C(=O)NCCC(O)C(=O)NCCCc1cncnc1)OC c1(C(N2C(CNC(=O)CCc3ccnc(Cl)c3)CC2)=O)ccc(O)c(CO)c1 C1(NC(C2(C(N)=O)CC2)=O)CN(C(C2CCC3C(C2)C3(F)F)=O)C2(CCC2)C1 CC(C)C(C#N)C(=O)N1CCCC(NC(=O)CCN(C)CCO)C1C c1(C(C)=O)cc(C(N2CC(O)(CNC(=O)Cc3ccon3)C2)=O)c(C)o1 CCCC(O)CC(=O)NCC1CN(C(c2cnccc2C)=O)CC1O c1(C(=O)Nc2ncc(CSc3ccc(F)cc3)s2)ccc2c(c1)COCO2 N#CC1(C(N2CC=C(CNC(C3CCC3)=O)CC2)=O)CC2C=CC1C2 C1(C(=O)NCCN(C)C(C2CCN(C)C2c2ccccc2)=O)CN2CCN1CC2 N1(C(c2cnn(CC)c2C)=O)CCCC(NC(=O)C(CN(C)C)N(C)C)C1C C(C)(C(=O)N1CC2CC1C2NC(c1ccsn1)=O)(C(C)C)OC C(C)(C)(CC(=O)O)NC(=O)NC(c1csc(C2CC2)n1)C C(=O)(C1CCCc2ccccc21)NCC(CCNC(C1(C)CC=CCC1)=O)OC N1(C(CCC(C)NC(C2(C)COC2)=O)=O)CC2OCCOC2C1 N1(C(CC2ON=C(CC)C2)=O)CC2=C(C1)CN(C(c1ccc(C(F)F)cc1)=O)C2 c1(N2CCCC(CC=C)C2)nc(=NCC2(c3ccccn3)CC2)[nH]c2ccsc12 Cc1cc(NC(c2ccc(C(C)F)cc2)=O)cc(C#N)c1 c1(NC(C(CCNC(CCCCOCC)=O)O)=O)ccc2ccoc2c1 CC1(C)C(=O)CC1C(N1CC(=C(F)CNC(c2ccc(-c3ccco3)[nH]2)=O)C1)=O N1(C(CCOCCCNC(=O)C(CO)C(F)(F)F)=O)CCCC12CCNC2=O N1(C(Cc2ccn(C)n2)=O)CC2(CC(NC(=O)C(C3CC(C)(C)CO3)O)C2)C1 C1(C(=O)NCC2(F)CN(C(C(C)(C)OCC)=O)C2)CCOC(C(C)C)C1 C1(C)(CC(N2CC(CNC(C(C)SC(C)C)=O)C2)=O)CC1(Cl)Cl N1(C(Cc2c(COC)cccc2)=O)CC2CCN(C(c3nnc(S)n3C)=O)C2C1 CC(C)CC(O)C(=O)N1CCC(CCC(=O)NC(C)CN2CCCCC2)C1 c1(OC)ccncc1C(=O)NC(C1(O)CCN(C(c2ccc(F)s2)=O)C1)C C(CO)(CCCCNC(=O)CS(=O)(=O)NC)NC(c1ncc(CC)nc1)=O c1(CNC(CC2(NC(CC(=O)NCC)=O)CC2)=O)ncccc1O CC(C)=C=CC(=O)NC1(c2cc[nH]c2C(=O)NC2(C)CCCC2O)CC1 c1(C(=O)NC2C(C)(C)CCCC2)n[nH]c2c1CN(C(=O)CCC1CCCOC1)C2 c1(NC(C)=O)cc(C(=O)NOCc2cn(C3C(C)CCCC3C)nn2)cnc1C c1(C(N2C(C(=O)Nc3cnc(OC)nc3C)CC3CC32)=O)c(Cl)cc(Br)cc1Cl n1(CC(N2C(CC)CN(c3ccccc3)CC2)=O)ccc(=O)c(O)c1C c1(C(=O)Nc2c(C(=O)NC(C=C)C)nccc2)cc(Cl)ncc1Cl C1(C)(NC(=O)Nc2cnn(C)c2C(C)(F)F)CCc2ccccc2C1 N1(C(c2c(CC)ncs2)=O)CCC2(CC2NC(c2nc(C)c(C)s2)=O)C1 C1(NC(c2n(CC)nnc2)=O)CCN(C(C2(C)CCCN(C)C2)=O)CC(C)(C)C1 c1(-c2nnc(N(CCNC(C)=O)CC)n2CC(C)C)c(F)c(F)c(F)c(F)c1F n1(CC(=O)NC(C)CNC(C2CC(C)(F)C2)=O)nc(C(F)F)cc1C1CC1 Cc1n[nH]c2cnc(C(=O)NC3CCOC(CNC(=O)Cc4ccco4)C3)cc12 C1(CNC(CCC=C(C)C)=O)CCC(C)CN1C(=O)CCc1ccn(C)n1 C#Cc1cc(C(=O)NC2COCC2NC(=O)CC2CCN(C)C2)ccc1C c1(CNC(C(=O)NCC(COCC)(C)C)=O)nc(C)c2c(n1)CCCC2 CC1CN(C(c2cocn2)=O)CCCN1C(=O)C(Cc1ccccc1)C(F)(F)F C=CCCCC(C(=O)NCC1CC1CCC)NC(=O)CC1(O)CCC1 C12(C(=O)NC3CC4CN(C(C5CC(C)(O)C5)=O)C3C4)CC3CC(CC(C3)C1)C2 N1(C(Cc2c(CC)cccc2CC)=O)CCOCC2(CCC2)C1 CC1CCC(CC(=O)NCC2(C(N)=O)CN(C(c3nnsc3N)=O)C2)OC1 C(=O)(N=c1cc[nH]c2cc[nH]c12)C1C2CN(C(c3cc(C)oc3C)=O)C1C2 C1(N(CCCO)CC(=O)N(CCCO)C)CNCC12CC2 C1(C(=O)NC(C(=O)NC)C2CC2)N(C(=O)C=C(C)C(C)(C)C)CCC1(C)C c1(C(N2CCC(C)(CCNC(C3N(C)CC(O)C3)=O)C2)=O)nnn2c1CCCC2 c1(C(=O)NCc2ccc(N3CCN(C(CC)=O)CC3)cc2)cc(F)ccc1Br c1(CCCC)ocnc1C(=O)N(CCCNC(=O)CCC1CCC1)C1CC1 n1(CC(=O)NC(CC)(C)CNC(=O)C(C)OCCC(C)C)nc(C)c(Cl)c1C c1(C(=O)NCCCCC(CO)NC(c2nc(C)oc2)=O)cccn2cnnc12 CC1CCN(C(c2ccc(F)c(Cl)c2)C)CC1NC(C1CCS(=O)(=O)C1)=O C1(C(N(CCCC(F)(F)F)C)=O)CC2CC1CN(C(C1CC(=O)NC(=O)N1)=O)C2 c1(OCC)cc(C)c(CNC2(c3nnnn3C)CCC3(CC2)CC3)cc1OC CC(C)(C)CCCC(=O)N1CCCN(C(=O)CN2CC(=O)NC2=O)CC1 CC1CCC(NC(C2CC(c3ccccc3F)C2)=O)CN1CC(N1CCOCC1)=O Cn1ncc(C2CC2)c1C(N1CC(=C(F)CNC(=O)Cc2csc(S)n2)C1)=O N1(C(C(COC(C)=O)C)=O)CCN(C(=O)C(O)CCN(C)C)CC1c1cnn(C)c1 O=C(C1=CCC(NC(C23CC2CNC3=O)=O)C1)NC1(C(F)F)CCC1 CC1=C(C(=O)N(C2CC(NC(=O)C(C)OC3CCCC3)C2)C)SCCO1 C1(C(=O)NC2CCCN(C(C(N3CCOCC3)C)=O)C2)CCc2ncsc2C1 Cc1nsc(NC2CC2)c1C(=O)NCC(C)CNC(=O)Cc1csc(S)n1 Cc1cc(F)c(C(=O)NCC2CCC2NC(=O)CN2OC(C)(C)CC2=O)c(F)c1 N1(C(CCOC2CN(C(CC(C)OC)=O)C2)=O)CC2C(N(C)C)C2C1 CS(=O)(=O)c1ccnc(NC2CC(NC(c3cnn[nH]3)=O)C2)n1 c1(C(C(=O)NCc2occ(C(=O)NC3(C(F)F)CCCC3)c2)O)ccc(Cl)cc1 c1(CNC(CCNC(=O)OC)=O)cc(C(=O)N(C(CO)C2CC2)C)no1 N1(C(C2C(CC)CC2)=O)CC(O)C(O)C1CNC(c1ccc(C2CCC2)cc1)=O n1(CC)nnnc1C(CCOCC1CC1)NCc1cc(COC)cs1 c1(CN(C(CSCCC)=O)C(C)C)c(F)c(F)c(C(F)(F)F)c(F)c1F c1(C(=O)NCC2C(NC(c3c(CC)nns3)=O)C2)csc2c1CCC(C)(C)C2 CC1(C)CCN(C(c2ccccc2)C(=O)NCc2ccc(F)cc2)CCS1(=O)=O Cn1ncc(-c2nn[nH]n2)c1C(N1CCN(CCCc2ccccn2)CC1)=O CC(C)(CCCNC(=O)CN1CCOC1=O)NC(C1CCCC(F)C1)=O C#Cc1ccc(NC(C2CCOC2CNC(C2(F)C(C)(C)C2(C)C)=O)=O)c(C)c1 c1(C(N(CCC(=O)NC(C2=NOCC2)c2nnnn2C)CC)=O)cnn(CC)c1 C(=O)(C(COC)CC)NCC1(F)CC(NC(C2(OCC)CC2)=O)C1 C(=O)(C1CCCc2ncccc21)NC(CNC(C1(CCCC)CCC1)=O)C(C)C C(=O)(CCCC(=O)NCCC1CCC(NC(c2cc(O)ncc2F)=O)C1)N(C)C c1(Cn2cc(CN3CC4CCCC(C)C4C3)nn2)ccc2[nH]c(=N)n(C)c2c1 C(=O)(C(CC(C)C)C(N)=O)NC1C2CN(C(c3noc(CC)c3C)=O)CC1CC2 C1(CNC(C(C(C)(C)C)C2CCC2)=O)CN(C(C2SCCS2)=O)CCC1(F)F N1(C(c2c(CC)noc2)=O)CC(NC(=O)CSc2nc[nH]n2)C(C(F)F)C1 c1(C(N(CC(CNC(c2cc(OC)c(F)cc2)=O)C)C)=O)c(F)ccc(O)c1O C(N=c1[nH]c2c(c(=NCCOC3(C)CC3)[nH]1)CCC2)c1ccc(C)cc1 c1(OCCCCNC(C(n2cc(CN(C)C)nn2)C)=O)cccc([N+](=O)[O-])c1 C12(NC(CSC)=O)CCCC1N(Cc1ccccc1)CC2 n1(CC(=O)N(CCCNC(C2CC(O)(CN)C2)=O)C)nc(C(F)F)cc1C1CC1 C1(CC(N2CCOCC(C(=O)NCCC3CC=CC3)C2)=O)Cc2ccccc2O1 C1(NC(C2CC(=C)C2)=O)COC2(CCN(C(=O)CCn3cncn3)C2)C1 C(=O)(CC1=CCN(C(=O)C=CCN2CCCC2)CC1)NC1C(C)COCC1 C1(C(=O)NCC2OCCCN(C(C3(SC)CC3)=O)C2)COc2cc(F)ccc2C1 c1(-n2ccc(NC(=O)C(=O)NC3COCC3N3CCOCC3)n2)ccccc1Cl C1(NC(=O)NCC(COC)(C)O)CC2CC1OC(=O)N2 c1(C(=O)NC(C(=O)NCC(CC(C)C)N(C)C)c2cccs2)cccc2[nH]ccc12 n1(C(C)C)cc(C(=O)NCCCCCNC(=O)COCC2CCCOC2)nn1 C12(C(N3CCN(C(c4nocc4Cl)=O)C(CCO)C3)=O)CC3CC1C2C3(F)F CC(C)C#CC(=O)N1CC(CC(C)NC(c2ccccc2)=O)C1 C1(NC(C=CCC)=O)CN(C(C2C(C=C(C)C)C2(C)C)=O)C(CC)(CC)C1 C1(C)(CNC(C2C(C)CC(C)O2)=O)CC(F)(F)CN1C(=O)CC12CCC(CC1)C2 C1(CNC(c2cc(OC)ns2)=O)CN(C(C2CC2F)=O)CC1O N1(C(C(CC)C#N)=O)CCC(NC(=O)Cc2ccc(F)cc2Cl)C2(CCC2)C1 c1(C(=O)NCC(CC)NC(C2CCCN2C(=O)NC)=O)nnn(C)n1 CCC(C)C(C)OC(=O)CNC(=O)C(=O)NCC(=O)SCCOC(C)C C(=O)(C(CC(C)C)CC(C)C)N1CCN(C(Cc2ccc(CC)cc2)=O)C2C1C2 c1(CNC(C(CC(=O)OC)C)=O)ccc(S(C)(=O)=O)[nH]1.C1CC1 Cc1cc(C(=O)NCC2CC2CNC(c2cc(-c3ccco3)[nH]n2)=O)cnn1 Cc1ncc(NC(=O)C(CN=[N+]=[N-])NC(=O)CNc2cccnc2)c(C)n1 C1(CC(=O)N(Cc2cnn(CCCl)c2)CC2CCCC2)CCC2CC12 C1(N(C(=O)COC2CC(CCO)C2)C)CCN(C(=O)COC(F)F)CC1 C1(NC(COCC=C)=O)CC2CCC(C1)N2C(c1ncn(C)n1)=O c1(CC)ccc(C)c(C(N2CCCC(C)C2CNC(=O)C(C)(C)OC)=O)c1 c1(CC)onc(C)c1CNC(=O)CCOCCCNC(C1(C#N)CC(=O)C1)=O c1(NC(c2scc(C(=O)Nc3cnc(C)c(Br)n3)n2)=O)cc(F)c(O)cc1Cl C(=O)(C(O)(C(F)(F)F)c1cn(CCC2CC2)nn1)N(C(C1CCC(=O)NC1)=O)CCO C1(CC(N2CCN(C(C(C)N(C(C)=O)C)=O)CC2C)=O)Cn2ccnc2NC1=O CC(C(C)(C)NC(=O)C(C)n1cnnn1)NC(c1cc(C2CC2)ns1)=O C1(NC(=O)Cn2ccc(C3CC3)n2)CC2(C1)CN(C(=O)C=Cc1ccncn1)C2 c1(-c2nc(C(C)SCC)nn2-c2ccccc2Cl)coc(S(N)(=O)=O)c1 Cc1cnccc1C=CC(=O)NC1CC(C)(CNC(=O)C(C)CO)C1 c1(C(C)C)cccc(F)c1C(=O)NCC12CC1CN(C(c1c[nH]c(=N)o1)=O)C2 CN1CC2C(C(=O)NC3(CNC(=O)CC4(C(F)(F)F)CNC(=O)C4)CCC3)C2C1 CC(F)CC(=O)NC(C)(CNC(=O)CCc1cnoc1)C1CC1 N1(C(c2cc(C)c(C(N)=O)cn2)=O)CC2CCC1CN2C(C1CCCOC1C)=O c1(C(=O)NC(COC)C(C)O)ccnc2c1CNCC2 C1(C(=O)NC2CCN(C(C(C(C)C)SC)=O)CC2)CC12CCCCCC2 C(=O)(N=c1[nH][nH]c2c1CN(Cc1cc[nH]n1)C2(C)C)c1c(OC)cc(C)cc1F C(=O)(C(C)(C)CC(F)F)NC1CCCN(C(CN(CCC#C)C)=O)CC1 c1(C(N2CCC2c2cn(CO)nn2)=O)cccn2ncnc12.c12ccc(cc1)s2 C(=O)(CCCN=[N+]=[N-])NC(CCCCNC(Cc1cccc(C)c1)=O)C Cc1cc(C(=O)NC2CCC2NC(c2ncoc2CN)=O)c2nc(C)n(C)c2n1 C(=O)(C1Cc2ccccc21)NCc1cccc(CNC(c2c(CC)onc2)=O)c1 C1(CC(N2CC(C)(CC)C2)=O)CC2(CC2)CN1C(c1ccc(Cl)o1)=O C1(CC(N2CC(N(C(=O)C(C3CC3)SC)C)C2)=O)(OC)COC1 C1(C(=O)NCC(CCOC)NC(=O)C(F)(F)C(F)F)CCCCS1(=O)=O N1(C(c2c(CC)csc2)=O)CC2CN(C(=O)Cc3cccc(C)c3F)CC2(C)C1 N1(C(CSCCOC)=O)CC(CC(=O)NCC(CO)CC(C)C)CC1(C)C C1(CNC(C=C(COC)C)=O)CCCC(NC(c2ccc(Br)cc2)=O)C1 C1(CCC)(NC(C2CC3(CC(OC)C3)C2)=O)CCCN(C(c2cocn2)=O)C1 C1(NC(C2(COC)CCC2)=O)CCN(C(c2ccc(Br)cc2OC)=O)CC1F C(C(C(F)(F)F)NC(=O)NCc1ccc(O)nc1)OC C(=O)(C1=C(Cl)CC1)NCC1(C)CC(NC(c2n(CC#C)ccc2)=O)C1 CC1CC(C)N(C(c2cccn2C)=O)CCN1C(=O)Cc1ccsc1 N1(C(CC(C)OC)=O)CCC2CN(C(=O)CCc3cncs3)CC2CC1 c1(C(N(CCCNC(Cc2c(C)ccs2)=O)C)=O)cnc(C(F)F)nc1 C1(CC(=O)NCC(CC)NC(C2(N3CCOC3=O)CC2)=O)CC2CC1C2 N1(CCCNC(c2cnn(Cc3ccccc3)c2)=O)CCc2ccccc21 N1(C(=O)CN2CCOC2=O)CC2(CCCC(CNC(C34CCC3C4)=O)O2)C1 c1(C(N2CCC(OCCNC(CC3C(CC)C3)=O)C2)=O)sc2ncccc2c1N C1(NC(c2ncn(C(C)C)c2)=O)C2CN(C(=O)CCc3ccncc3)CC12 CON(C)C1CCN(C(C2CCC2NC(c2cccc(C)c2F)=O)=O)CC1 c1(C(=O)OCC)nc(C(=O)NCC(C)NC(=O)CCN2CCCCC2)cs1 n1(C(=O)NC2CCCC(O)C2O)ncc(S(=O)(=O)N2CCOCC(CC)C2)c1C C1(CNC(c2cc(C)ns2)=O)CCC2(CO1)CC(NC(=O)CC(C)(C)C1CC1)C2 N1(C(CC2(C#N)CCOCC2)=O)C2CCCC1CN(C(=O)CCCCC1CC1)C2 CC(C)CCC(O)C(=O)N1CCC(NC(C2CCC(C(F)(F)F)CC2)=O)CC1 Cc1cc(C)c(CC(=O)Nc2ccc(Cl)c(N(C)C)c2)c(C)c1 C1(NC(c2c(OC)cccn2)=O)CC2CC(NC(=O)CCc3cc(Cl)cs3)CC12 C1(NC(COCCC#C)=O)CCCN(C(c2cnn(C)c2C(F)(F)F)=O)CC1F N(C1CCCc2cc(F)c(F)cc21)C(c1c(N)cncc1Cl)=O Cc1cn(CC(=O)NCC2(NC(C3CC(=O)CO3)=O)CCCC2)c2ccccc12 N1(C(CNC(CNC(=O)OC)=O)=O)CCN(C(=O)C(C)C)CC1C C1(C(N(CCCO)CC#C)=O)(NC(=O)CC2CCC3CC23)CCN(C)C1 Cc1cc(C(N2CCC(c3ccccc3)(C(N)=O)C2)=O)c(F)c(Br)c1 c1(OC)cc(COC(=O)C(N2CCCCC2)C)cc(F)c1O Cc1cc(C)c(C(=O)NCC2CCCN2C(=O)CCc2ccccc2Cl)c(C)n1 N1(C(C2COCC(C)O2)=O)CCC2(CCN(C(c3cc(O)ccc3Cl)=O)CC2)C1 CC1CN=C2NC(C(=O)N3CC(N(C)C(c4cc(C(C)(C)C)no4)=O)C3)=NN2C1 C#CC1(C)CCCN(C(=O)C(C)(C)C(C)NC(C2CCN(OC)CC2)=O)C1 N1(C(C=CC(=O)N(C)C)=O)CC(F)CC1CN(C)C(C1(O)CCCC1)=O N1(C(c2n(CC)ncn2)=O)C(CNC(=O)CN2CCN(C)CC2)CC2COCC12 CC(C)CC(CNC(=O)CCCCCNC(C1(CC2CC2)CC1)=O)CO c1(C(=O)Nc2onc(C)c2Br)cc2ccc(-c3cnn(CC(C)(C)O)c3)cn2c1 N1(C(CS(CC)(=O)=O)=O)CC23CCCC2(C1)CN(C(C1CCOC(=O)CC1)=O)C3 Cc1cc(N2CCN(C(c3ncccc3F)=O)CCC2C)ncc1[N+](=O)[O-] N1(C(C2CCCC(O)C2)=O)CCC=C(C(=O)N2C(CO)CCC23CCC3)C1 C1(NC(CCSCC)=O)CN(C(c2cc3cccnc3o2)=O)C2(CCCOC2)C1 c1(N2CCN(C(CCC#C)=O)C3C2C3)cc2ncnn2cn1 N1(C(C(C)Oc2ccccc2)=O)CCCCC(NC(c2ccc(C(N)=O)o2)=O)C1 N1(C(=O)CCc2ccc[nH]2)CCC2CCN(C(C34CC5CC3C4C5)=O)CC12 Cc1nc(O)c(C(=O)NCCc2cnc(NC(C3CCN(C)CC3)=O)s2)nc1C c1(C(N2C3(CC(CN(C)C)C3)CC2)=O)nc2c(Br)cncc2[nH]1 N1(CC2C(CNC(C(CC3CN(C(c4n(C)ncc4)=O)C3)F)=O)C2)CCCOCC1 N1(CC(=O)NCC(CCNC(c2cc(COC)[nH]n2)=O)O)CCCCC1=O Cc1noc(C)c1C(C)Nc1nccc(N2CC(CO)C(O)C2)n1 Cc1cc(C(N2CC(CNC(=O)Cn3ccnn3)CCC2C)=O)cc(C)c1 C(C)(C)(C(C)CC(=O)NCC(C)C(=O)OCC)NC(c1cc(CC)oc1C)=O c1(C(=O)NC2CCCCC2NC(C2CCCC23CCC3)=O)cc2n(n1)CCCC2 C(CCCC(=O)NCCOCCOCCC1CCSC(C)C1)OCC N1(C(C(C(C)(C)C)CO)=O)CCC2CCC(C1)N2C(=O)CCOC1CC(F)(F)C1 c1(C(c2n(CC(=O)NCC)nnn2)NCCN(C)C)c(OC)ncnc1OC C(C(=O)NCC1CCCCN(Cc2coc(C)n2)C1)(C(C)(C)C)NC(C)=O C1(NC(c2nc(C)c(C)s2)=O)C(C)CN(C(c2ccc(Cl)cc2F)=O)CC1C N1(C(C(c2ccccc2)C)=O)CCC2(CCCC2C(N2CCNCC2(C)C)=O)C1 N1(C(c2ncn(CC(=O)OC)c2)=O)CCC2CC12C(=O)NCC1(O)CC(CO)C1 c1(C(=O)NCCC(C)N(C(c2c(OC)cccn2)=O)C)c(C)nc2sc(C)nn12 C1(CNC(c2n(CCC)ccc2)=O)CC(N=c2[nH]c3cc(Br)ccc3o2)C1 c1(NC(C2(C)N(C(C(C(C)C)O)=O)CC2)=O)cc(Cl)ccc1C#N N1(C(C(=O)OCC)=O)CCC2(CC1)CCN(c1ncc3ccn(C)c3n1)CC2 NC1CC2CCCC(C1)N2C(=O)NCCOc1ccc(Cl)c([N+](=O)[O-])c1 C(=O)(C(F)(F)CC1CCCO1)NCC1CCN1C(C1(C)CCCS1)=O c1(C(C)O)ccccc1N1CCCC1.C1(N)CN(CCc2ccncc2Cl)C2CC12 C1(CN(C(=O)Cc2c[nH]nc2O)C)CN(C(C2CCN(C)C2)=O)CCO1 C(CN=c1[nH]c2c(c(=NCCCS(C)(=O)=O)[nH]1)CC(C)CC2)C1CC(C)C1 CCCCCC(F)C(=O)N1CCC(CCNC(c2ccncc2F)=O)C1 CCC(C)(C(=O)NCc1c[nH]nc1C(=O)NC1CCC(C(=O)NC)C1)OC c1(SCC)cc(CCNC(=O)CC2(C)CCN2C(=O)C(CC)N(C)C)on1 CCC(CC(F)(F)F)C(=O)NC1CCCN(c2ncnc(C)c2Br)C1 c1(C(C(=O)N2CC(C(C(=O)N3CCC3CF)N(C)C)C2)(C)C)ccc(F)cc1F.CO N1(C(c2cccc(C)c2)=O)C2CCC(C(N3CCCC3(C)C)=O)C1CC2 c1(OC)ccc(C(=O)NC2CC(CNC(=O)CCc3ccncc3)C2(C)C)nc1 c1(C(N2CC(C(C)NC(C(=Cc3cccs3)C)=O)C2)=O)cc2c[nH]cnc-2n1 C(=O)(CC(C)CCC)N1C(CC)C(C(=O)NCC(O)COC(C)C)C1 C=CC1(C(N2CCCC(CCCO)C2)=O)CCN(C(=O)Cc2cc[nH]c2)CC1 C1(CC)C(NC(=O)COCC(N2CC=CC2)=O)CCCN1C(c1ccns1)=O C1(C(=O)NC2(CC=C)CN(C(=O)C(C)CCOC)C2)CCOC(C)(C)C1 c1(OCC)ccc(C(=O)NCCCN(C(c2ccnnc2C(C)C)=O)CC)cc1 N1(C(=O)COC2CC=CC2)CC23CCCC2(C1)CN(C=O)C3.C1CCCCO1 c1(C(=O)NCCCC(C)NC(C(C)(C)OC(C)=O)=O)cc(C2CC2)cc(F)c1 Cc1cc(C(N2CCCC(C)(CNC(c3cc(C)n(C)c3)=O)C2)=O)ccc1O CCC(CC(=O)NCC1CC(OC)CN1C(c1cn(C(C)(C)C)nn1)=O)C(F)F C1(CNC(c2ccno2)=O)CC2(CCN(C(=O)C(F)n3cccn3)CC2)CO1 N1(C(C2(CC=C)CC2)=O)CC(CNC(=O)Cc2ccno2)C(O)C1 C1(C(=O)NC(COC)(C)C2CC2)CN(C(=O)Cc2cnccn2)CCO1 C1(NC(CC2C(CNC(CC#N)=O)C2)=O)CCOCC1 CC1(C)C(NC(=O)C2=CCCC2)CC1CNC(c1conc1-c1ccccc1)=O c1(CC(=O)NC2C(NC(COCc3cc(C)no3)=O)C2)cc(C)sc1C C(=O)(C1=CC(O)CCC1)N1CC(NC(c2c(CC)n(C)nc2)=O)C2(C1)CC2 CN1CCCC(F)(C(=O)NCCC2CCCN2C(=O)CCCn2cccc2)C1 CCC(C)(C)C(O)C(=O)NCC1(C)CCCN1C(c1cncnc1C)=O CC(C)(CCNC(C1CCCC1O)=O)C(=O)Nc1ccc(F)c(O)c1 N1(C(C(N2CCCC(OCC(=O)OC)CC2)=O)=O)CCSC2(CCC2)C1 c1(C(N2C(CN(C(=O)COC3(C)CCC3)C)CCCC2)=O)cc2ccccc2[nH]1 C1(C)(C(=O)NC2CC(CC(=O)N(C)CC3(CC(C)C)CC3)C2)CC(F)C1 C1(O)(CNC(C(CSC)OC)=O)CCCN(C(c2sccc2F)=O)C1 C(C(C(=O)N1CCC(NC(c2cnccc2Cl)=O)C1)C(C)(C)C)OCC=C C1(OC)CN(C(=O)CC(C)(C)N2CCOCC2)CC1NC(C1(O)CCC1)=O C(=O)(CC(C)(O)C=C)NC(CC=C)CNC(c1ccc(N(C)C)nc1)=O Cc1nn(C)c(=O)c(C(=O)NC2COC3(C2)CN(C(=O)C(O)C(F)(F)F)C3)c1C c1(C(=O)NCCN(C(C(C2CCOC2)OCC)=O)C)ccc(N(C)C(C)C)nc1 C(=O)(CC(F)(F)CC(=O)NCC(C)(C)CN(C(=O)C(C1CCOC1)OC)C)OC c1(C(C)NC(Cn2cc(CCCOC)nn2)=O)ccccc1[N+](=O)[O-] N1(C(C2C(C)CC=CC2)=O)CCCN(C(=O)CC2CCC(C)(C)O2)CC1CO N1(C(C(CC)c2ccccc2)=O)CC2CC(NC(=O)C(COC)N(C)C)CC1C2 C(=O)(CC(CN(C)C)CC)NCC(CCCC)NC(c1c(C)nsc1Br)=O c1(OC)ccnc(C(N2CCC(C(C)NC(=O)CC3CC4(CC4)CO3)C2)=O)c1F c1(CC(=O)NC2CC(N(C(Cc3cc(C)no3)=O)C)C2)cccc2cnccc12 C(=O)(CS(=O)(=O)c1ccccc1Cl)NC(CN(C(CC(CCCC)O)=O)C)CC Cc1nsc(C(=O)NC(CCNC(C2CC(C)CO2)=O)C(C)C)c1N C(=O)(C(F)(F)C(O)C(C)C)NCCN(C(=O)Cc1cccc(OC)n1)CCOC c1(OC(C)C(=O)NC2CCN2C(=O)CCOCCCCC2CC2)ccccc1F C1(CNC(c2ccc(O)nc2)=O)CN(C(C2(F)CCCC2)=O)CC2(CCC2)O1 Cc1c(C(=O)NCC2CC2CNC(=O)CC(=O)N(C)C)oc2ccc(Cl)cc12 c1(NC)ncccc1C(=O)NC1(CC(=O)NCCC2CCCCCC2)CCC1 c1(C(=O)NCCC2CC(NC(=O)C(O)CC3CCCC3)C2)cc2cccnc2s1 c1(CCN=C(NC(C2CCOCC2)C)NCc2cscn2)nc2c(s1)CCCC2 CC(C(C)(C)C(=O)NC1(C2CC2)CCOC1)NC(=O)COCC1CCCC1 c1(C(N2CCOC(CC)C2)C(=O)NCC=C)cc(Cl)c(F)c(Cl)c1 Cc1cc(F)cnc1C(=O)NCC(O)C(=O)N(CC(C)(O)C1CC1)C c1(C(N2CCC(=C)C2)C(=O)NCC)ccc(C)c(C#N)c1 C1(NC(CCCCC#C)=O)CC12CCC(NC(=O)Cn1ccc(C(F)F)n1)CC2 CC1(NC(C2CC23CC(NC(=O)CCCN=[N+]=[N-])C3)=O)CN2CCC1CC2 c1(C(=O)NC(C2C(C(N(CC(O)CO)C(C)C)=O)C2)C)ccnn1C Cc1c(C(=O)NCC2(C(C)(C)O)CN(C(=O)C(C)N3CCC3)C2)ccn1C1CC1 c1(CCC(=O)NC2CCN(C(C(CO)NC(N)=O)=O)C2)ccccc1Br c1(CCC)cc(C(=O)NC(C)C(C)NC(=O)CCCC(=O)OCC)cc(O)n1 CC1CCCN(C(c2cnn(CCF)c2)=O)C1CO.c12cccc(n1)CNC2=O c1(OC)cc(F)ccc1C(N1CCC(O)(C(=O)Nc2cc3ncsc3[nH]2)C1)=O N1(C(c2n(C)nc(O)c2)=O)CCCC(CNC(=O)C(C)(F)CC2CCCC2)CC1 CC1CC(NC(c2nc(C(F)(F)F)ccc2N)=O)CN(C(C2(C3CC3)CC2)=O)C1 Cn1c(C(=O)NC2CCN(C(=O)CC3CCC4(CCC4)O3)C2)cc2occc12 C1(O)(C)CN(C(C2CC2(C)C)=O)C1.N12CC(C1)C(=O)N2.CC(C)(C)OC1CC1C N1(C(CC2CCC(=O)N2)=O)CCCCC(NC(=O)C=Cc2cccs2)CC1 c1(C(=O)NCC#CCNC(c2cn3ccsc3n2)=O)ccc(C(F)(F)F)c(Cl)c1 c1(C(N2CC3CCCC2C3)C(=O)NCCCC2CC2)ccc(F)c(C(F)(F)F)c1 C(=O)(NNC(=O)c1ccc(OCC(N)=O)cc1)c1nc(CC)[nH]n1 CCC(CCCC(=O)NC1(CC(N)=O)CCC1)NC(c1cnn(C2CC2)c1)=O c1(C(N2CC(NC(c3c(CC)cco3)=O)C(C)C2)=O)nc(C)c(C)nc1O c1(-c2cc(C)on2)cc(Cl)cc2c1NCCC2 N1(C(C2N(C(Cc3nc(C)oc3)=O)C(C)C2)=O)C2CCCC1CC2 c1(-c2cn(C3(O)CCN(C(C(CC)C)=O)CC3)nn2)oc2ccccc2c1C c1(C(=O)NCCOCCNC(C(C)(C)c2ccsc2)=O)ccc(Cl)cc1 C1(NC(CCCCN(C(C)C)C)=O)CC(C)CN(C(C23CCCC(CO2)C3)=O)C1 c1(OC)ncc(-c2cn(CC(=O)N(C)C)nn2)cn1.c12cc(nn1C)C(=O)NC2 c1(C(=O)NC2CC23CC(NC(c2nncs2)=O)C3)cc2c(s1)CCCC2 CC1=C(C(=O)NCc2ccoc2C(N(C)CP(C)(C)=O)=O)COCC1 c1(C(=O)NC2C(NC(=O)Cc3ccc(O)cn3)CC2)nnc2n1CCCCC2 Cc1c(O)c(=O)ccn1CC(N1CCC2(NC(=O)CCc3cc[nH]n3)CC2C1)=O C1(CCC)(NC(=O)CN(C2CCSC2)C)CCCN(C(C2(Cl)CC2)=O)C1 C1(C(N(CC(COC)O)C)=O)CCCCCCN1C(=O)CC1CCCCC1O N12CCC(CC1)OCCC(C)(C)N1CCCC1C2=O.c1(O)cccnc1.CC CN(C)S(=O)(=O)N1CCCCC1c1nc(CC23CCC(CN)(C2)C3)no1 c1(CC)ccc(C(=O)NC2CCCC2C(=O)NCCC2CCCC2)nc1 N1(C(C2C(N(c3scc(CC)n3)C)COC2)=O)CCN(C)C(C2CCCCC2)C1 C(C(C(C)C(C)C)NC(=O)C=C1CC1)NC(CNC(c1ccc(C)s1)=O)=O c1(CC)ccc(NC(=O)C(=O)NCC2CCCS2(=O)=O)c(C(=O)OC)c1 N1(C(c2c(CC)ncs2)=O)CCC(C)(CCNC(C2(C)CCCS2)=O)CC1 C(=O)(CC1=CSC2=NCCN12)NCC(C)NC(=O)CC1CCCOC1 N1(C(C2(C#C)CCC2)=O)CCCC(NC(=O)C(c2ccccc2)SC)C1 C1(CC(=O)NC2C=CCN(C(C3CCSC3)=O)C2)CCCC12CC2 c12cc(ccc1C)NC(=O)N2.c1(COC)ccnc(C(=O)NCC(F)(F)F)c1 CCCCCCCCCn1cc(C2CC(O)CN2C(=O)C(C)(O)C(C)C)nn1 C12(NC(C(F)OC)=O)CCCN(C(=O)C(C)=C3CCCC3)CC1C2 C(=O)(C(F)C(F)(F)F)NCC1CN(C(C(=O)NCCNC(C)=O)=O)C(C)C1 c1(OC)ccc(OC(C)C(=O)NCC2CCN(C(c3nc(C)sc3C)=O)C2)cc1 CC1CCN(C(=O)NCc2scnc2NC(=O)OC(C)(C)C)C1 Cc1c(Br)ccnc1C(=O)NCCN(C(c1cnnc(O)c1)=O)CC1CC1 c1(C(N2CCC(CNC(C(P(C)(C)=O)O)=O)(CO)CC2)=O)cnc2[nH]ccc2n1 S(=O)(=O)(c1ccc(F)cc1)N1CC2CN(C(c3c(O)cccc3Br)=O)CC21 c1(OC)cccc(CC(=O)NCC2CC2CNC(C2CC2C=CCSC)=O)c1 C#Cc1cc(C(=O)NC2CC3CCC2N(C(=O)CC(O)CC)C3)cc(F)c1 N1(C(c2cc(C)c(N)cn2)=O)CC2CC3CC2C1C3NC(=O)Cc1cc[nH]n1 C(=O)(C(F)C(C)(F)F)N1CCC(CC=C)(C(=O)NCCC2C=CCC2)C1 CCCC(CCC)CC(=O)N1CCCN(C(C2CCCCC2F)=O)CC1 Cc1cc(CCC(=O)NC2CCN(c3nccc(Br)n3)CC2CO)cc(C)c1 c1(OC)cc(N)ccc1C(=O)NCCC(C)N(C)C(C12CCCC(CO1)C2)=O CN=c1[nH]cc(C(=O)NC2CCN(C(=O)C(C)(c3ccccc3)N(C)C)CC2)o1 C1(C(=O)NCCCCCC#C)C2CCCC2CN1C(=O)C(O)CN(C)C c1(CC(=O)N(C)CC2CCN(C(C(CC#C)C)=O)CC2)cc(Cl)ccc1O C1(NC(CC)=O)CCN(C(=O)C=Cc2cccs2)CC1C C1(N(C(c2n(C=C)nnc2)=O)C)CCCCN(C(=O)C(C)OCC)C1 C1(NC(=O)Cc2cnc[nH]2)CC2CCC1C(NC(C1(CCF)CCOCC1)=O)C2 Cc1nn(C)c(Cl)c1C(=O)NCC#CCNC(C1(Cl)CC1)=O c1(OC)ccc(SCC(=O)N(C)CC2(O)CCN(C(C3CNC(=O)N3)=O)C2)cc1 c1(C(=O)NCC(n2cc(CC(=O)O)nn2)C)cc(N2CCCC2)nc(Cl)c1 c1(OCC)ccc(-c2nc(C)c(C(=O)NC3(CC(=O)OC)CN(C)C3)s2)c(F)c1 c1(-c2cc(NC(=O)CC34CCCN3CCC4)sc2)cccc2scnc12 C1(C(=O)OCc2cccc(C(N)=O)c2)CCc2nc(-c3ccccc3)ncc2C1 C1(C(=O)NC2CCCCN(C(C3(C#C)CCCC3)=O)C2)CC2(C1)CC(F)(F)C2 N1(C(Cc2cc(C)sc2)=O)CC2(C1)SCCC2NC(c1cc(C(F)F)ncn1)=O Cc1cc(C(c2ccccc2)Oc2cc(Br)ccc2C)nc(C)n1 CC(C)(C(=O)N1CC(c2cn(CCN3CC3)nn2)(CO)C1)C1CCCO1 c1(C(C(=O)NC(C(=O)N(CCCOC)C)C)O)cncn1C C1(C(=O)NC(C)(C)CC(=O)N2CC(C)(C)C2C2CC2)CC12CCOCC2 N(C(=NCCCF)NC1CCCn2nc(C)nc21)CC(COC)C N1(C(CC=C)=O)CCC2(COC(CNC(c3cc(C)c(C)c(F)c3)=O)C2)C1 C1(F)(C(=O)NCC2C(C(N3CC(NC(=O)NC)C3)=O)OCC2)CCCCCC1 c1(OC)ccc(Br)c(C(=O)NCCCCNC(c2ccn(C)c2C)=O)c1 CC1(C)COC(C(=O)NCC2(C(C)(C)O)CN(C(=O)Cc3ccc(F)cc3)C2)C1 c1(CNC(CC2ON=C(C)C2)=O)cccnc1CNC(c1nc(C)n(C)n1)=O C1(C(N2C(CN(C(CC=C)=O)C)CCC2)=O)(C(=O)OC(C)(C)C)CCSCC1 C1(NC(CCNC(=O)OCC)=O)CC(C)N(C(C2CC3CC3C2)=O)C1 C1(O)(CNC(COC(C)=O)=O)CCCN(C(C2CCN(C(C)=O)CC2)=O)C1 CCC(CC)CC(=O)N(CCC(C)NC(=O)Cn1ccnc1C)C C1(C(F)(F)F)(OC)CC(CNC(=O)C(C)O)(NC(=O)Cc2cnc[nH]2)C1 C(CCF)(C(=O)NCCCc1nc[nH]n1)NC(c1ccc(O)nc1)=O Cc1cnccc1C=CC(=O)NC1(CN(C)C(C2(C)CCCC2O)=O)CC1 C(=O)(C#CC1CCCOC1)N1CCCN(C(c2ccc(C)cc2O)=O)CC1 c1(C(N(CCCNC(=O)CC2CCC(F)(F)C2)C(C)C)=O)ccc(F)cc1C#N C#Cc1cc(F)ccc1CNC1(OC(C)=O)CCN(C(=O)CSC)CC1 c1(C(=O)NCC2N(C(C3ON=C(CC)C3)=O)CC2)cnc2cc(C)ccn2c1=O CCC(CC)(CO)C(=O)NCC(C)(C)OCC(N1CC2(C1)CC(C)(O)C2)=O c1(C(CNC(=O)CSC)NC(CCSCCCC)=O)cn(C)nn1 C#CC1(O)CC(C(=O)NC(C2CCCCC2)C(C)NC(C2CC3CC3C2)=O)C1 c1(SCC(N2C3C(CNC(C4(CC=C)CCC4)=O)C(C3)C2)=O)cc(F)ccc1F C(=O)(C(CC(C)C)NC(=O)OC(C)(C)C)NCCCN(C(CC(C)C)=O)CCO CCC(CC)(CCNC(c1cc(C2CCCC2)no1)=O)NC(=O)C1CC1 C(=O)(C1=CCc2ccccc21)NC1CN(C(c2c(=N)[nH]nc(Cl)c2)=O)C1 N1(C(c2onc(C)n2)C)CCC(C2CCCN(C(=O)C(C)C3CC3)C2)C1 N1(C(C2OCCN(C)C2)=O)CCC(C2(NC(=O)CCS(C)(=O)=O)CC2)C1 c1(OC)cc(Br)cc2c1CN(C(=O)NCCC1CCCC(C)C1)CC2 C(C(=O)NC(C1CCCN1C(=O)CNC(c1ccccc1)=O)C)(C(C)C)OC c1(C(=O)NCCC(C)N(C(C2(C(=O)OC)CC2)=O)C)ccc(C(F)(F)F)nc1C c1(C(N2CCN(C3C(NC(C(C=CC)O)=O)CCC3)CC2)=O)cnc(O)c(F)c1 C1(NC(C2CSC2)=O)(CF)CCN(C(C2(C(F)(F)F)CC2)=O)C1 c1(C(=O)NCCCC(C)NC(c2coc(CO)c2)=O)ncncc1F C1(C(N(C2CCN(C(=O)C(c3cccc(C)c3)C)C2)CC)=O)CC(N=[N+]=[N-])C1 CC1CN(C(c2csc(-c3cnccn3)n2)=O)CC1NC(C1CC(N(C)C)C1)=O c1(C(N2CC(CNC(=O)CCOC3CC3)OCCC2)=O)cnc2ccsc2c1 C(N=c1[nH]c(N2CCN(c3cncnc3)CC2)nc(=N)[nH]1)C1(C)CC2CC2C1 c1(NC(C2C3CN(C(C(CC=C)(F)F)=O)C2C3)=O)cnc2cc(Br)ccc2c1 Cc1ccccc1C(N1CCN(CC2CCCN(C(c3cnco3)=O)C2)CC1)=O C1(n2cc(CC(C(C)C)O)nn2)CCCCNC1=O.C12CCCCC1CNC2=O C1(C=C)(C(=O)NC(C#C)C)CCN(C(c2cc(Cl)cs2)=O)CC1 c1(C(=O)NCC(CNC(CS(CC)(=O)=O)=O)O)cccc2ccncc12 N1(C(CC2CCC(C)O2)=O)CCC(N(C(=O)COCC2(F)CC2)C)CC1 c1(CCC(=O)NCC2(NC(CSCC=C)=O)CCC2)cc(Cl)no1 C(=O)(C1=C(Cl)CCOC1)NC1(CNC(C2C(C)C(=O)C2)=O)CC1 CC(C)(CC(F)(F)F)C(=O)NC1CCN(C(c2ccc(Cl)nc2)=O)CCC1CO c1(C(=O)NC(CC)CNC(=O)Cc2cncc(F)c2)cnn2c1CCCC2C c1(C(=O)NC2(CC)CCN(C(=O)C(F)=C(C)C)CC2)cccc(S(C)=O)c1 CC(C(=O)NC1CCCCN(C(=O)C(c2ccc(Cl)cc2)(C)C)C1)C1=CCCC1 N1(C(c2cc(OC)ncn2)=O)CC2CCN(C(C3COC4COCC4O3)=O)C2C1 C1(CCN(C)C(C2CCCC2CNC(c2csc(O)n2)=O)=O)CCOCC1 C1(N(C(c2c(C)ccs2)=O)C)CCN(C(C2CCCSC2)=O)CC1 c1(NC(C2CCCN(Cc3cc[nH]c3)CC2)=O)cc2nccn2cn1 N1(C(C2(OC)CCSC2)=O)CCC(C(=O)NC(C2CCC2)C)(C(C)C)C1 c1(-n2c(C)ncc2)ccc(C(=O)NCCCC2(NC(=O)C(=O)NC(N)=O)CC2)cn1 C(=O)(C1=Cc2ccccc2OC1)N1CC2CCN(C(CCSC)=O)CC21 N1(C(CNC(CC(C)C)=O)=O)CCOC(CN(C)C(c2cc(F)n(C)n2)=O)C1 C12(C(N(CCC(=O)NCC3(O)CCSC3)C3CC3)=O)CSCC1C2 C1(NC(C(CC)(C)OC)=O)CCC2CCN(C(c3ccoc3Cl)=O)C1C2 N1(C(C(CC)CC)C(=O)NCCN2CCOCC2)CCCC2(CCN(C)C2)C1 C1(CNC(C2N(CC)CCOC2)=O)CN(C)CCN1C(=O)Cc1ccc(Cl)cc1 C1(CNC(COCCC)=O)CCCC2(CN(C(c3cc(C)ccc3Cl)=O)C2)O1 c1(CN(CCc2ccsc2C)CC)c(F)cc(Br)cc1F.SCC N1(C(Cc2n(C)nnc2)=O)CC(C(N2CCOCC(CO)C2)=O)C2(CC2)C1 C=C(C)CC(C)C(=O)NCC1CCN1C(c1cc(-c2ccccc2)c[nH]1)=O C1(OC(c2c(C)cc(F)c(F)c2)=O)CCn2c(C)nnc2C1.C1(=O)CNC(=O)N1 S(=O)(=O)(c1ccc(N2C3CCC2c2ccccc23)c(Br)c1)NC1(C)CC(C)C1 CC(C)CC(F)C(=O)NCCC(C)(C)NC(=O)CCOCC=Cc1ccco1 C1(O)(CNC(c2sccc2F)=O)CCCN(C(=O)CNc2ccccc2Cl)C1 c1(C(N(CCCNC(=O)C(C)n2cccn2)CC)=O)cccc(C(C)(C)C)n1 S(=O)(=O)(c1ccc(C#N)c(NCC2CN3CCN2CC3)c1)NCCN(C)C N1(CC(=O)NCCCC2(NC(C3C(C)(C)C3C(F)F)=O)CC2)CCC(C)(O)C1 C(=O)(C(C)CC(C)(F)F)N1C(CN(C(c2c(C)[nH][nH]c2=N)=O)C)CCCC1 CC1CCNCCC1N(C(=O)CN1CCOCC1)Cc1cccc(F)c1F n1(CC(=O)NCC(CNC(c2c(C)cccc2Cl)=O)C)ncc2ccccc12 N1(C(CSC)=O)CC(CNC(c2cccc(-c3ccsc3)c2)=O)OC2CCCC12 N1(C(CCC(=C)Cl)=O)CCCCC(NC(C2CC2(c2ccccc2F)C)=O)C1 c1(C(N(C(C)(CO)C(=O)N2CCN(C(C)(C)C)CC2)C)=O)cc2cccn2cn1 c1(C(N(CCCNC(C2CCC3C2C3(F)F)=O)C(C)C)=O)ccn2nnnc2c1 C1(CNC(C2(S(N)(=O)=O)CC2)=O)CC(F)(F)CN1C(=O)C=CI CC(C)C(CNC(c1cnn(C2CCCC2)c1)=O)NC(C1CCCC1O)=O c1(N2CCCCC(SC)C2)nc(NC2CC(CO)(CCl)CC2)c2ncsc2n1 C(=O)(C(C)CS(C)(=O)=O)N1C(CNC(=O)CCc2ccccc2Cl)CC(OC)C1 C1(C(=O)NC(C(C)NC(=O)CCOCC2CCCO2)C)CCN(C)CC1 c1(NC(C(C)OC(C2CCCOCC2)=O)=O)ccc(C(C)(C)C)cc1 c1(C(=O)NCCC(C)NC(c2c(OCC)nccc2)=O)cc2ccc(C)cn2c1 O=S(=O)(c1cnc(N2C3CCC2CC(O)C3)c(Cl)c1)NCc1ccncc1 N1(C(C2(CC)CCCC2)=O)CC(NC(c2cc(OC(F)F)n(C)n2)=O)CC(F)C1 c1(C(=O)NC2C(O)CCN(C(c3cn(C)nc3)=O)C2)ccn2c1CS(=O)(=O)CC2 c1(CCC(=O)N(C2CCN(C(c3n[nH]cc3C)=O)C2)CC)cncc(F)c1 c1(N2CC3C(C2)N3C(C2CN(C)C2)=O)ccc2nc(C)nc(COC)c2c1 Cc1ccc(C(=O)NC2CN(C(C3CC(CF)C3)=O)CC2(C)C)c(F)c1F C1(NC(C2(c3ccc(C#C)cc3)CCC2)=O)CCN(C(C2(C)CC2)=O)CC(O)C1 c1(NC(C)Cc2ccc(C(F)(F)F)cc2)ccc2c(c1)CN(C)CCC2.C(CC)S CN1CCCCC1C(=O)NC1CC(CC(=O)NCCCCCCC2CC2)C1 c1(C(=O)NC2C3(CC(NC(COCC#C)=O)C3)C2)nc2cccnc2s1 c1(NC(C2CC(Nc3cc(OC)ncn3)C2)C)ccc(OC)c(F)c1 CC(=O)C(C)(C)CC(=O)NC(CO)C(=O)NCCCCCCCO C1(CC(C)NC(C2(C)CS(=O)(=O)C2)=O)CCN(C(=O)CSC(F)F)CC1 C(=O)(C1Cc2ccccc21)NCC1C(C)(C)N(C(=O)CNc2cccnc2)CC1 C(=O)(CCS(=O)(=O)c1ccccc1)NC(CN(C)C(C1CC12CCC2)=O)(C)C c1(C(N2CCC(C(N3CC(O)(CC=C)C3)=O)C2)=O)c[nH]ccc1=O c1(OC)cc(C(F)(F)F)nc(N2CCCC2C2CCN(C(=O)C=CC(N)=O)C2)n1 C(=O)(CS(=O)c1ccc(Cl)cc1)N1CCC(CC#C)(C(=O)N(CC)CC)CC1 C(CC(C)C)(CS(=O)(=O)N)OC.N1(CCC2CCCC2c2ccccc2)CCN(C)CC1 N(C=CC(=O)C(F)(F)F)C(C1CCC2(CN(C(=O)C(Cl)(Cl)Cl)C2)O1)=O Cc1cc(C(N2CCC(C)C2CNC(=O)C(C)(F)F)=O)nc(N(C)C)n1 C1(NC(C(OC)OC)=O)CN(C(=O)CCOCC2CCCO2)CC12CCC2 C1(C(=O)OC)CCCN(C(c2ccc(SC)cc2)C(=O)NCC#CC(=O)OC)C1 N1(C(Cc2cnc(C)s2)=O)C(CNC(=O)CC2CCC(O)C2)CC2COCC12 C(=O)(CCCc1nc(C(C)C)no1)NC(CNC(C1C(C=C)C1)=O)CC C1(CC(C)C)(C(=O)NCC2(COC)CC2)CCCN1C(=O)CCc1cnccn1 C(C(C)C)(C(O)C(=O)N1CCCC(C)(NC(C2CC(O)C2)=O)C1)OC CCCC(C)(CCC)C(=O)N(CCNC(c1ccc2cc(C)oc2c1)=O)C1CC1 C1(C(C)(C)NC(C2C=CCS2)=O)CCN(C(=O)C(O)CN2CCCC2)C1 NS(=O)(=O)C1(C(=O)NCC2CCC2NC(c2n[nH]c3c2CCSC3)=O)CCCC1 CCC(CCOC)C(=O)N1CCCCC1CCC(=O)NC1CCCN(O)C1=O Cc1ccc(C(C)(C)C(=O)NCCN2CCN(C(c3coc(Cl)n3)=O)CC2)cc1 N1(C(CC=CCC)=O)CCC(CC(N2CC(c3ccccc3)C2)=O)C1 C=C(C)C(F)(F)CC(=O)NOCc1cn(CCCc2ccccc2)nn1 C1(C(N(C2CCC2)CC#C)=O)CC12CCN(C(=O)C1=CCN(C)C1)C2 c1(CC)cc(C(=O)N(C2CCCN(C(=O)CC3COCCN3C)C2)C)cc(O)n1 C(=O)(CCc1ccc[nH]1)OCC1C(CCC)C1 c1(C2C(C(N(C(C)CNC(C3CC(O)C3)=O)CC)=O)C2)ccccc1 c1(C(=O)NC2C3CN(C(Cc4cn(C(C)C)nn4)=O)CC32)cc2ncccc2[nH]1 c1(C(=O)NC(CNC(c2cnc(CC)[nH]2)=O)(C)C2CC2)ccc2sc(=N)[nH]c2c1 C(CC(C)C)(C(=O)NCC1CC2CN(C(=O)C=Cc3cocn3)CC12)NC(C)=O C(=O)(CCCCCNC(C1CCNC1=O)=O)N1CC(CC(C)C)C1 N1(C(CCOC)=O)CCCC(C2CCCN(C(C3(CO)CCC3)=O)C2)C1 c1(C(=O)NCCC2CCN(C(CC(C(=C)C)OCC)=O)C2)nccn2ccnc12 c1(NC(CC(CCC)NC(C2CC23CCC3)=O)=O)cc(F)c(O)cc1C N1(C(c2cnnc(Cl)c2)=O)CC2CCN(C(=O)Cc3ccccc3O)C2C1 Cc1cc(C)c2nc(N3CCC(C4(NC(C5CCCN5C)=O)CC4)C3)sc2c1 c1(C(=O)NCCCN(c2ncnn3cccc23)CC)ccc2c(c1)CCCO2 c1(C(=O)NCC(C)N(C(c2nc(C)ccc2F)=O)CC)nsc2ccc(C)cc12 c1(O)ccc(Cl)cc1Cl.C1(CC#N)CCCC1NCCCCN CC(C)CC(C(=O)NC1CC(NC(=O)C(C)(C)c2ccn(C)n2)C1)C(N)=O c1(C(=O)NC(C(=O)NCc2cc(CC)[nH]n2)CC2CC2)cc(C#N)cn1C C1(CNC(CC(=O)OC)=O)CN(C(=O)CN(C)C2CC2)CCC1C(F)(F)F C(=O)(C(O)CC[S+](C)C)N1C(CCN(C(=O)C=C2CCCCC2)C)CCCC1 C(=O)(CCC(=O)N1CCCCC1C(C)NC(C12COCC(C1)C2)=O)N(C(C)C)C CCC(CCC(=O)NC(CC)C(N)=O)NC(c1cnc(C)c(C)c1)=O C1(NC(c2ccc(-c3cn(CC(=O)O)nn3)o2)=O)CCCCCC1O C1(N(C(C2N(C(C)=O)CC(O)C2)=O)C)CC2CC1N(C(=O)CC(C)(F)F)C2 C1(C#N)(C(=O)NC(CSCCCOC)C(=O)O)CC(F)(F)C1 CCC(C)(O)C(=O)NC(CNC(c1ccc(C2(C)CC2)cc1)=O)C(C)C C1(NC(c2c(C)nc(CCC)s2)=O)CCC2CN(C(=O)CC(C)C3CC3)CC2C1 c1(C(=O)NC2C(NC(=O)CCF)COC2)n[nH]c2ccccc12 Cc1scc(C(N2CCC(NC(c3cc[nH]c(=N)c3)=O)C2)=O)c1Br C12(C(=O)NC3CN(C(CN(C)CC)=O)CC4C3C4)CCOC1CC(=O)NC2 C(C1CCCc2sc(C)nc21)NC(NCC1CC(SC)C1)=NCC(C)C N1(C(C2C(C)C2)=O)CC2(CCC(CNC(=O)COCC3CC3)O2)C1 C1(O)(CC(=O)NCCCCCNC(=O)CSCc2ccccc2Cl)CCCCC1 N1(C(c2cn(CC=C)nc2)=O)CCC(CNC(C2CC(C)C2(C)C)=O)(OC)CC1 C1(CNC(c2cc(CNC(COC(C)=O)=O)sc2)=O)CC(=O)N(C)C1 N1(C(c2cc(C)sc2-n2cccc2)=O)CC2CC(NC(=O)Cc3cnoc3)C1C2 Cc1cccc(F)c1CC(=O)NCC=CCNC(C1CN2CCC1C2)=O N1(C(C)=O)CCC(C(N2CCC(CCNC(C3(S(N)(=O)=O)CC3)=O)C2)=O)CC1 N1(C(=O)CCSc2ccccn2)CCC2CN(C(C3OCCCO3)=O)CCC2C1 C1(CNC(C(CC)C)=O)CC2(C1)CN(C(c1ccsc1SC)=O)C2 N1(C(C=CC)=O)CCN(C(c2cnc3sccn23)=O)C(CF)C1 c1(NC(C2CCC(CNC(C3CCCO3)=O)CC2)=O)cc([N+](=O)[O-])ccc1Cl N1(C(c2cc(C)c(F)cn2)=O)CCCN(C(=O)Cc2nncn2C)C(C)C1 CCC1=C(C(=O)N(CC(C)NC(c2ccc(C(C)(C)C)nc2)=O)C)SCCO1 C#CCCCCC(=O)NC1CCN(C(=O)COc2ccc(Br)c(C)c2)C1 C1(C(=O)NCCC(=O)NC(CC)C)CN(C(c2csc(C)c2)=O)CC12CC2 C1(C(=O)NC(C(=O)N(CC)Cc2cn(C)nn2)CO)CCCCN1C c1(-n2cc(C(C(C)(C)OCC)NC(C)COC)nn2)ccccc1OC(F)F C1(NC(c2c(CC)con2)=O)CC2CC1N(C(=O)C=Cc1cnn(C)c1C)C2 C1(OC)CC2(C1)CC(C(N1CCC(C(C)NC(=O)C(CO)C(C)C)C1)=O)C2 CC(C)C(CNC(c1csc(C(F)(F)F)n1)=O)NC(c1ncoc1C1CCC1)=O CC1(C)C2CCC(C(=O)NCC3CCCN(C(=O)C=C4CC4)C3)C1C2 c1(C(C(=O)NC(CNC(C=COCC)=O)C(C)(C)C)O)c(C)cccc1C CC1CCOCC1C(=O)N(CCNC(C12CC(C1)C2)=O)C1CC1 c1(COCC)nc2c(s1)CCN(C(c1csc(NC(C=COC(C)=O)=O)n1)=O)C2 Cc1cccc(C=CC(N2CC(CN(C)C(c3occc3C3CC3)=O)C2)=O)c1 CCCC(C(=O)NC(C)C(C)(C)NC(=O)C(O)C(C)C)OCC C(=O)(CCC(F)(F)F)NCC(=O)NC(C(=O)OC)C1CC1 C1(N=c2ccc3nnnn3[nH]2)(CNC(CN2CC(=O)NCC2)=O)CCC1 N1(C(c2cc(O)cc(F)c2)=O)CC2CCN(C(c3c(F)cccc3I)=O)CC2C1 c1(CNC2CC(NC(=O)C=Cc3ccco3)C2)cccnc1O c1(C(=O)NCC2C(NC(=O)Cc3cncs3)CC2)cnc(O)s1 c1(NC(C(CC=C)C)c2nnnn2CC2CCCO2)ccc(OC)c(C)c1 O=C(COCCN)NNC(=O)CNC(c1ccc(Cl)s1)=O C1(CC=C)(C(=O)NC2(CSC)CC2)CCCN1C(=O)C(C)CCOC c1(OC)cc(F)cc(C=CC(=O)NC2CCN(C(=O)CC(C)(C)C#N)C23CC3)c1 n1(CC(N2CC(NC(C(c3ccccc3)NC(COC)=O)=O)C2)=O)cnc(Br)c1 n1(CC)cc(CC(=O)NCCN(C(c2ccnn2C(C)C)=O)CC2CC2)nn1 C1(C)(NC(c2ccc(COC)o2)=O)CCN(C(=O)C(C)N(C)C)C1 c1(C(N2CCC(C(C)(C)NC(c3c(C)nsc3)=O)C2)=O)cc(F)cc(F)c1 Cc1ccc(C2CC2C(N2CCC(F)(c3ccc(C(F)(F)F)cc3)C2)=O)cc1 c1(C(=O)NCC(C2CCC2)NC(CSC(C)C)=O)cccc2cc(Cl)ccc12 C1(NC(C2(CCOC)CC2)=O)CCCN(C(c2nnc(C)s2)=O)C1 Cc1cc(C)c(C(N2CCN(C)CC2CNC(=O)C(O)P(C)(C)=O)=O)cc1C CC(C)(C)CCCC(=O)NCC1OCCC1C(N1CCC2C(O)CC12)=O c1(OC)cccc(C(O)C(=O)NC(C2CC(NC(=O)C(C)(C)OC)C2)C)c1 CC(C)C(C#N)C(=O)NCCCC(C)NC(=O)CC(=O)Nc1ccc(F)cc1 C1(C(=O)NC(CCCC)CNC(=O)C(C)(C)F)CC2CCC(C1)N2C(C)C c1(OC)ccc(C=CC(=O)NC23CC2CN(C(C2CC4(CCOC4)C2)=O)C3)cc1 C1(O)(CNC(CS(=O)(=O)NC)=O)CCCN(C(=O)CCc2cnc[nH]2)C1 Cc1ncc(C(N2CCCC(C(C)(C)NC(=O)C(=O)NC(C)C)C2)=O)cc1N CC1=C(C(=O)NCC(C)(CO)NC(=O)Cc2cc(C)cc(F)c2)CCS1(=O)=O N1(C(c2c(CC)cns2)=O)CCCCC1CCN(C(=O)C(F)=C1CCCC1)C N1(C(Cc2nc(C)oc2)=O)CCC(C)(C)C1C(=O)NC1(C(C)O)CC1 N1(c2cc(NCc3n(CC)cnn3)nc(C(F)(F)F)n2)CCC2(CCCCC2)C1 C1(NC(c2cnn[nH]2)=O)CCN(C(=O)CCCc2cc(Cl)sc2Cl)CC1O CCCCC(CC)C(C(=O)NCC(C)C)N(C(C)C(C)C)C C(=O)(C1CCc2nccn21)NCC(C(C)C)(F)C(=O)N1CCC12CCCCC2 Cc1cccc(C(=O)NCC=CCNC(=O)COC2CCOCC2)c1O CC(CC(C)NC(c1cnn(C2CCCC2)c1)=O)N=c1ccn2c(Br)cnc2[nH]1 c1(C(N(C(C2CCOCC2)C)C)=O)c(CNC(C2CCCC(=O)N2)=O)cnn1C CC1(C)CCOC1C(N1CC(O)(C(F)C(=O)NCCCc2cnccn2)C1)=O c1(CNC(CCc2ccc(C(=O)Nc3cn(C)nn3)[nH]2)=O)cc(Cl)c(F)cc1F C1(C(=O)NCC2N(C(C(C)OCCC(C)C)=O)CCC2)CCOC(CC(C)C)C1 Cc1[nH]nc(C(N2CC(CF)(NC(C3CCCC(O)C3)=O)C2)=O)c1C C=CC(C)(O)C(=O)N1CCC(O)(CNC(c2cc(Cl)c(Br)s2)=O)C1 C1(NC(C(C)OCC(F)(F)F)=O)CC2CC(NC(=O)C=Cc3cc[nH]n3)CC2C1 C1(C)(C(N2CCC(C)(NC(Cc3c(C)ccnc3)=O)CC2)=O)COC(C)(C)CO1 C#CCN(OC)C(=O)C(c1ccoc1)NC(c1csc(C#N)c1)=O c1(C(=O)NCC(C2CCCCC2)NC(C2C(C)C2)=O)cc([N+](=O)[O-])cnc1N N1(C(CSCCC)=O)CC23CCCCC2(C1)CN(c1cc(OC)nc(OC)n1)C3 c1(C(N2CCCN(C(CC(=C=C)C)=O)C(CO)C2)=O)cc(C)nc2c1CCCC2 Cn1nc(I)cc1S(=O)(=O)NC(C1CCC2(CC(CO)C2)CC1)=O CC(C)CC(CC(=O)NCC1CCN(C(C2(C)CS(=O)(=O)C2)=O)CC1)CC(N)=O N1(C(c2cccc(OC)c2)=O)CC(C)N(C(c2oc(C)cc2C)=O)CC1C S1(=O)(=O)c2ccc(cc2Cl)N1.c1(SCC(C)C)ccc(C(N)=O)cc1Cl.C1CS1 C1(C(=O)NC(C)(C)CNC(C2CCC2(F)F)=O)CC2(C1)CC2(F)F c1(OC)ccc(C(CC(=O)O)NCCc2nnc(C)s2)cc1OC N1(C(C2CC(NC(c3c(C)nn(C)c3N)=O)C2)=O)CCc2n[nH]cc2C1 c1(OC)ccc(CO)cc1C(=O)NCCCC(C)NC(=O)CC1(C)CCCO1 c1(SCC(N2CC(NC(C3CC4C(C)(C)C4C3)=O)C(O)C2)=O)ccc2c(c1)CCC2 O=C1NC2(CCN(C(C3C4CCN(C(C5(O)CCOC5)=O)CC34)=O)C2)CO1 c1(CC(=O)NC23CC(CNC(CCOC)=O)(OC2)C3)coc2ccc(F)cc12 c1(C(=O)NC2C(NC(c3c(C)nc(CC4CC4)o3)=O)C2)cc(N)nc(Cl)c1 C1(C(=O)NC(CC=CC)C(=O)OCC)CC2(C1)CC1(CCC1)C2 C(=O)(N=c1[nH][nH]c2c1CN(Cc1cccc(I)c1F)C2)c1c(C)ccs1 N1(C(C(C(CC)C)O)=O)CCn2ncc(S(C)(=O)=NC(=O)C(C)CC)c2C1 C(=O)(C(O)C(C)(C)CC)N(CC(CO)(CO)NC(C(CCC)F)=O)C c1(C(C)(C)C)cc(C(=O)NOCc2ccccc2)ccn1.C1(CCF)C(=O)N1 N12C3CCC1CN(C3)C(=O)c1cc(ccc1Cl)NC(=O)C2CC=CC.c1(OC)ccccc1 c1(C(=O)NCC2CCN(C(C3(CF)CC3(F)F)=O)CC2)coc2c1CS(=O)(=O)C2 c1(N(CC(O)CF)C)ccn2ncc(S(=O)(=O)NCCc3ccncc3F)c2n1 C(C(C)(C)CNC(=O)C(F)(F)Sc1cnn(C)c1)N(C(C1CC(CCC)C1)=O)C Cc1nn(C)c2sc(C(=O)NC3CCN(C(c4cc(F)cs4)=O)C3C)cc12 C1(CCCC)CCC(NC(=O)C(N2CCC(COC(C)(C)C)C2)=O)CC1 C(=O)(C(CNC(=O)COCCCN(C)C)CC1CCCC1)NC(CC=CC)CO c1(C(C)NC(=O)NCC2(C(F)(F)F)CCCCC2)cc(F)cc(F)c1 C1(NC(c2c(CC)cno2)=O)CCCC12CCN(C(C1CCCC1O)=O)CC2 c1(CC(=O)NC2CC(C)(NC(COCC#C)=O)C2)nn(C)c(=O)c2ccccc12 C(CC(C)(C)C)(C(=O)NCCc1ccnc(O)c1)NC(CC1C(C)C(=O)CC1)=O C1(NC(=O)CN2CCNC2=O)COC2(CNC(=O)C(F)F)CC1C2 CCCCC(C(=O)N1CC2CCN(C(c3cnc(C)[nH]3)=O)CC12)C(C)C C1(C(=O)NCCCCNC(CCC(=C)C)=O)CCCC(=O)N1C c1(C(N2CCN(C(C(c3c(C)cccc3)C)=O)CC2)=O)cn2c(C)cccc2n1 C1(C(=O)NCC(CCC)C)CC(O)CN1C(=O)C(C(C)O)N(C)C C(=O)(CCCC(=O)N1CCC(C(C)(C)C)(CNC(=O)C(C)OC(C)(C)C)C1)OC c1(NC(=O)OC)ccc(C=CC(N2CCN(C(=O)C=CC(C)(C)C)CC2)=O)cc1 c1(C(N2CC(CCNC(C3(SC)CCC3)=O)OCC2)=O)cncc(Cl)c1C N1(Cc2ccc(S(C)(=O)=O)cc2F)CCC2(CC(O)CNC2=O)C1 C1(C)(CNC(c2nn(C)c(C3CC3)c2)=O)CCCN(C(C23CCC(C2)OC3)=O)C1 C1(N(C(CN(C)C(=O)C2CC2)=O)C2CC2)COC2(CCCC2)C1.C1CC(=O)N1 N1(C(C)CCNC(=O)NCc2ccoc2)CCCCC1CN(C)C N1(C(Cc2cc(C)on2)=O)CCOC2(CCN(C(c3cc[nH]c3)=O)C2)C1 c1(C(=O)NC2CC3CN(C(CCN(CC)CC)=O)C2C3)csc2c(O)ccnc12 C(C)(CO)(C(=O)N1CCC(CCC(=O)NCCC2CCCC(C)C2)CC1)OC N1(CC(=O)Nc2[nH]c(=N)sc2-c2ccccc2)CCC2(CC1)CC(F)CO2 CCCCCC(CC)C(=O)NCC1CCC12CCN(C(c1ocnc1C)=O)CC2 N1(C(CCCOCC)=O)CCC(C)C(CNC(C23CCC(CC2)O3)=O)C1 CCCCC(O)C(C)C(=O)NCC1CC2CN(C(=O)C(c3cnn(C)c3)=O)CC12 C1(C(=O)NC2C(CNC(c3ccc(Cl)cc3)=O)CCC2)CC2CCC(C1)O2 c1(C(=O)NCC2=CCN(C(C3C(C)(CC)C3)=O)CC2)csc2ccc(C)cc12 N1(CCn2cc(CCOC(C)=O)nn2)CCN(C(=O)CCCC2CCCC2)CC1 C1(C(=O)NC2C3(CN(C(c4c(C)cns4)=O)C3)CCC2)CC(F)(F)CCC1(C)C C1(CNC(Cc2ccn(CC)n2)=O)(NC(c2csc(C)n2)=O)CCCCC1C Cc1cc(C)c(CCN=c2[nH]c(CN3CCC(CO)CC3)cs2)c(C)c1 c1(C(=O)NC2(CO)CCCN(CC(COC)O)C2)sc2ccccc2c1Cl C1(NCCCCCN(C(C)=O)C(C)C)CC2(CCOC2)CO1 CC1(C(=O)NCC2CC2NC(C2(C)COCCO2)=O)Cc2ccccc2C1 c1(C(N2C(C)CN(C(=O)C(C)(O)C3CC3)CC2)=O)cc2c(ccn2C)s1 n1(CC)nnc(C(=O)NCCNC(=O)Cn2cncc2C(=O)OC)c1C C1(CNC(c2c(CC)n(C)nn2)=O)CCCCN(C(c2cncs2)=O)C1 Cn1ncc(C2CCC2)c1C(N1CC2C(CNC(c3ccc(O)cn3)=O)C2C1)=O C=CC1(C(=O)Nc2cnc(F)nc2)CCN(C(c2nonc2C)=O)CC1 C(c1ccccc1OC(F)(F)F)=CC(=O)N(C1CCCN(C(=O)C2CC2)CC1)C C1(CNC(C(C)OCCC=C)=O)CCCCC1C(=O)NC1(CCO)CCC1 CCC(C#N)C(=O)NCCC1CCCN(C(c2ccccc2SC(F)(F)F)=O)C1 CN1CCn2[nH]c(=NC(=O)C3CCCCC3n3ccnc3)cc2C1 C1(C(C)C)CN(C(C2CN(C)C(=O)N2)=O)CCN1C(C1CC(=O)N(C)C1)=O Cc1cnc2n1CCCC2C(=O)NC12CCC(CC1)N(C(C1SCCCS1)=O)C2 C1(C(N(CCNC(C2C(C(F)F)C2(C)C)=O)CC)=O)Cc2cc(Cl)ccc2O1 C1(C(N2CCC(CC(F)F)C2)=O)CCN(C(=O)C(F)C2CCCC2)C12CC2 c1(C(=O)NCC(CCOC)NC(=O)C(C)C(C)C)csc2c1CCCCCC2 C1(C(N2C3CC(NC(=O)Cc4cc(Cl)cc(Cl)c4)(C3)C2)=O)CCc2nccn2C1 Cc1[nH]c2ncnc(NC3CCC(NC(C4CC4(C)C(C)C)=O)CC3)c2c1C c1(C(C(=O)NC(CN(C(C(C)OC)=O)C)C)C2CCCC2)ccncc1 c1(C(N2CC3C(CNC(CCc4cc(C)on4)=O)(C3)C2)=O)c([N+](=O)[O-])cnn1C c1(C(C)C)cccc(NC(c2cc(CNC(C3CCCN3C=O)=O)on2)=O)c1 CC1(C)CCCCN(C(=O)CC2(NC(C3CCCCCC3)=O)CC2)C1 N1(C(C(CC)=CC)=O)CC2(CCOCC2)CC1CNC(=O)C(C)CC(F)(F)F c1(C(=O)NCC(CCCC)NC(=O)C(C)OCCC(C)C)cc(C)cc(C)n1 Cc1c(C(=O)N(CC(C)CNC(C2(F)CC=CCC2)=O)C)cncc1Br CC(=O)CCCC(=O)NCC(c1cccc(C)c1)NC(c1cc(=O)cc[nH]1)=O C1(CC=C)N(C(c2cc(OC)c(C)cc2Br)C(=O)NCC2CC2)CCCC1(C)C C1(CNC(CS(C)(=O)=O)=O)CCC2(CN(C(=O)CCC=Cc3ccccc3)C2)O1 C(CCCCCC(=O)NC1CCc2nncn2C1)NC(=O)CC1CC(C2CC2)C1 N1(C(C(CC)SC)=O)CC(N(C)C(c2cc(N)cc(F)c2)=O)C2(CC2)C1 c1(CNC(CC(C)(C)NC(CC(=O)NCC)=O)=O)cccc(C)c1F N1(C(c2ccc(SC)s2)=O)CCOC(CCNC(=O)C(N2CCC(C)C2)=O)C1 Cc1ccc(C(=O)NC2CN(C(=O)Cn3cc(C#N)cn3)CC2C)nc1 CC1=C(C(=O)NC(C)C(CO)NC(c2[nH]c(C)nc2C)=O)Cn2ncnc2N1C C1(CNC(CSC)=O)CCCN1C(=O)C(C)(F)c1ccccc1 c1(C(NNC(c2c(C)ccc(OC)c2)=O)=O)cc(S(C)(=O)=O)cc(C(F)F)c1F CCCC(CCC)CC(=O)NC(C)(CNC(C1(F)CCC(=O)CC1)=O)C1CC1 C1(C(=O)NC(CCCC)C)C(C)OCCN1C(=O)Cc1ccc(F)nc1 CCCCC(CNC(C1C=CC=CC=C1)=O)NC(c1c(OC)noc1C)=O c1(C(N2C(CCNC(CC(C(C)C)C)=O)CCC2)=O)ccc2nc[nH]c2c1F c1(C(N(CCC)CCNC(=O)CSCCC(F)(F)F)=O)cccc(F)c1NC C1(C(C)NC(c2cc(Cl)cs2)=O)CN(C(c2cn(C3(CO)CC3)nn2)=O)CCO1 c1(C(=O)NCC2CC(OC)CN2C(=O)C(C)(F)F)cccc2nc(C)nn12 N1(C(c2n(C)c(O)nc2)=O)CCC2CCN(C(=O)CCC(N)=O)C2C1 Cc1nn(C)cc1CC(=O)NC(C)CCCNC(=O)CCOCCN(C)C c1(C(=O)NCC(CNC(C2(C#N)CCCOC2)=O)O)cc2ccccc2o1 Cc1cnc(CNC(=O)Cc2cccc(C)n2)c(C)c1 C(=O)(CCC(C)(C)C)N(CCC(N1CC(C(N(C)C)=O)C1)=O)C Cc1c(S(=O)(=O)NC(C(C)(C)C)c2nnnn2C2CC2)oc2ccc(F)cc12 CC(C)CCN=C1NCC2CC2C(C2CC2)N1.c1(NS(C)(=O)=O)ccc(SC)cc1 c1(C(=O)NCC(CNC(C2(C)CCCC2(F)F)=O)F)nc[nH]c2ncnc1-2 CCCCS(=O)(=O)NCC(=O)NCC1(F)CC(NC(=O)CC(=O)OC)C1 c1(C(=O)NC(C(=O)NOCCCO)C2(O)CCC2)cnc(S)nc1 C1(NC(C2CCCC(C(F)(F)F)C2)=O)(CO)CCN(C(=O)Cc2cc[nH]n2)C1 C1(NC(C(C2CCC2)OC)=O)CCC2CN(C(c3ccc(C#N)s3)=O)CC2C1 CC(C)(COCC(F)F)C(=O)N1CC(C(N)=O)(CNC(=O)CN2CC3CC3C2)C1 Cc1cc(F)c2cc(C(=O)NC3CCN(C(C4CCSCC4)=O)C(C)C3)[nH]c2c1 C1(CCC)CN(C(=O)C(C(C)C)OC)CCN1C(c1cnc(C2CC2)nc1)=O C=CCC(CNC(C1CCO1)=O)NC(c1cnc(C(C)C)o1)=O C1(CCn2cc(C3(F)CN(C(Cc4cnc(C)o4)=O)C3)nn2)CCS(=O)(=O)C1 CCC1=NOC(CC(=O)NCC(CC)NC(C2CCN(c3nccs3)CC2)=O)C1 C=CCC(C(=O)NCCC(C)CCNC(C1CCC(=O)N1C)=O)C(C)C Cc1nccc(CNC(c2ccc(C3(O)CC(N)C3)cc2)=O)n1 N1(CC)CCOCC1CC(N1CC(CO)(NC(=O)C(c2cnn(C)c2)OC)C1)=O C1(NC(c2c(C)cn(C(C)C)c2)=O)CCN(C(=O)CSc2nncn2C)CC1C C1(CNc2cc(OC)nc(OC)n2)CCCC2CCCCC12 c1(C(=O)NC2C(CNC(CC34CC(C)(OC3)C4)=O)C2)ccc(Cl)c(C#N)c1 N1(C(c2cn(CC=C)nc2)=O)CCC(C=C)(C(=O)N2CC(C)(O)CO2)CC1 N1(C(CC2(NC(C)=O)CC2)=O)CCCN(C(c2[nH]nnc2C2CCOC2)=O)CCC1 N1(CCNC(c2scc(C)c2Cl)=O)CCCN(C(C2(C#N)CC(C)C2)=O)CC1 CC1(C)CC(=O)N(C(=O)NCC2(CNC(C3(F)CC3)=O)CC2)C1=O O=C(CCCCC1CC1)NCCCN1CCN(C(c2ccc(Cl)o2)=O)CC1 C1(NC(C(N)=O)=O)CCCCC1NC(=O)CC1(C(F)F)CC1 c1(OCC(N2C3C(NC(CC4C(C)=NNC4=O)=O)C(C3)C2)=O)ccc(F)c(Cl)c1 C1(C(N2CC(OCCNC(=O)CC34CC(C3)C4)C2)=O)CC2CCC1C2 C(CC1CCCCC1)(C(=O)N1CCC1COC1CCCO1)C(=O)OC(C)(C)C C1(NC(C(C)SC)=O)CC2(CCN(c3cc(C)c(C(N)=O)cn3)C2)C1 C1(N(C)C(C2(C#N)CC2(C)C)=O)CN(C(=O)CCC(F)(F)F)CC1(C)C CCC(CC(F)(F)F)NC(C1COCCN1C(C1(N2CCCC2)CC1)=O)=O c1(C(CNC(CC=C)=O)NC(=O)CC2CCNC(=O)C2)cccc(Cl)c1Cl N1(C(C(C)OC)=O)CCN(C(c2cc3occc3[nH]2)=O)C(c2ncc[nH]2)C1 c1(C(=O)NC23CC(NC(c4cccc(F)c4)=O)(C2)C3)cccc2c1CNC2=O C1(CC=C)(C(=O)NC2COC(C(C)C)C2)CN(C(=O)CCOC(C)=O)C1 C#CCC(C)(C)CNC(C1CSCCN1C(C1CC(C)=NO1)=O)=O c1(C(=O)NC2CN(C(C(CC)(C)F)=O)CC2CC(C)(C)C)cnn2cccnc12 C1(C(=O)NC23C(CN(C(CCc4cc(C)nn4C)=O)C2)C3)CN(C)CCN1C N1(Cc2ccc(COC)o2)CC2C(C1C(=O)Nc1cccc(O)n1)C2(C)C N1(C(c2c(OC)n[nH]c2)=O)CCC(O)C(NC(=O)CC2CC3(CC3)CO2)C1 C1(NC(C(C(=O)OC)C)=O)CCCN(C(c2cnn(C(F)(F)F)c2)=O)CC1 C(=O)(C(C(C)C)N1CCCCC1)NC1C(NC(c2c(SC)snn2)=O)C1 Cc1cc(CCNC(=O)C(c2ccccc2)NC(C2(F)CC=CCC2)=O)nn1C c1(OC)csc(C(=O)NCC2CN(C(=O)CC3CC3(Cl)Cl)C2)c1OC N1(C(C(CCSC)O)=O)CC2(CCC(NC(=O)CCCC(C)O)CC2)C1 C1(C(N2C(C)(C(=O)OC)CC2)=O)CNC(=O)CN1C(=O)Cc1cc(C)no1 C1(C(=O)NC(c2nc(=O)o[nH]2)C)CC=CC(NC(C2CCC(=O)NC2)=O)C1 CC1(CCCO)CCCN1C(C1OCCC1NC(=O)CC12CCC(CC1)C2)=O c1(CC)ccc(CNC(=O)C(=O)N(CC(F)CC)C(C)C)nc1 Cc1ccccc1C(C)C(=O)NCCCCCCNC(C1CC(F)(F)CS1)=O c1(CC)[nH]nc(C(N2CC(n3cc(Cn4cc(C)cn4)nn3)C2)=O)c1Cl CCCCC(O)CC(=O)N1CCN(C(c2cn(C)c(C)cc2=O)=O)CC1CCO C1(CNC(CC2(OC)CCC2)=O)CCN(C(=O)CC2CCCC2C)C1(C)C C1(C(C)NC(CNC(=O)OC)=O)CCCCN1C(C1(C(F)F)CCCC1)=O C(=O)(NNc1c(F)cc(F)cc1I)C12OCC(NC(=O)OC(C)(C)C)C(C1)C2 c1(NC(C2=NOC(C)C2)=O)nc2c(s1)CC(F)(F)CC2 N1(C(CCOCC#C)=O)CCOC(CNC(=O)CC2CCC(OC)CC2)C1 CCCCC(=O)Nc1c[nH]nc1C(=O)NCCOCCOC N1(C(C(C2CCOC2)OC)=O)CC(NC(C2CCCC2)=O)C2(CCOCC2)C1 C1(N(C(c2c(OC)csc2)=O)C)CCN(C(c2cc(C(C)(C)C)on2)=O)CC1C N1(C(COCCC#C)=O)CC(NC(=O)CNS(=O)(=O)N(C)C)CC12CCOC2 C12(CNC(C3N(CC)CCC3)=O)CC(CN1C(c1cccc(CC#N)c1)=O)C2 c1(C(N2CC=CC(NC(c3c(C)oc(C4CC4)n3)=O)C2)=O)nnn2c1CSCC2 Cc1ccc(O)c(C(=O)NCC2(F)CC(CNC(=O)C(C3CCCCC3)C)C2)c1 N1(C(C(CSC)C)=O)CC(NC(c2cncc(N(C)C)c2)=O)C(SC)C1 C1(C(=O)NC(C2CCOC2)CNC(c2ccn(C)n2)=O)CCC2(CC1)CC2(F)F C(CCCCCCCO)=CC(=O)NCCC1C(C)CN(C(C2(F)CCCC2)=O)C1 C(=O)(C1=C(C)OCCS1)NC1CCCCN(C(c2cn(CC)nn2)=O)C1 C(=O)(C1=CCC(C)(C)CC1)NC1CC(C)N(C(c2cn(C)[nH]c2=N)=O)C1 C#Cc1ccc(C(=O)NC(C(=O)O)C(O)Cc2ccccc2)nc1 c1(C(=O)NCC2N(C(C(N)=O)=O)CC=C2)ncnc2c1ncn2C1CC1 C1(C2CN(C(=O)CCCN3C(=O)CCC3=O)C2)(NC(=O)C(O)CN2CCC2)CC1 c1(OCCC(CN(C(=O)Cc2ccccc2C(F)(F)F)C)OC)ccc(Cl)cc1 C#CCC(C)(C(=O)NCCC(CCC)C1CC1)NC(C1CCOCC1(C)C)=O N1(C(C2C=CC(NC(c3c(C)nn[nH]3)=O)C2)=O)CCN2CCCCC2C1 Cc1cc(C(N2CC=C(C(=O)NCC3CC34CCOC4)C2)=O)nc(O)n1 C(c1cccc(F)c1)=CC(=O)NCC1COCCN1C(=O)CCCc1cccs1 N1(CC(=O)NCC2CC2NC(c2cn(CCC3CCC3)nn2)=O)C(=O)CCC1=O C1(C(=O)NC(C)C#N)CC(O)CCN1C(=O)C(N)=O C1(Cn2cc(C(C)(O)C(=O)O)nn2)CN(C(=O)Cc2csc(C(F)F)n2)CCO1 c1(NC(C(C)NC(Cc2cc(CC)no2)=O)=O)cccc(Cl)c1O c1(OC)ccc(S(=O)(=O)N(C(=O)Cc2cccs2)CC2(O)CNC2)cc1 C1(CCNC(c2nnnn2C2CC(F)(F)C2)C2(CC)CC2)NC(=O)NC1=O c1(NC(C(=O)NC(C2CCOCC2)CC)=O)ccc(C)cc1 N=c1[nH]cc([N+](=O)[O-])cc1C(=O)NC1(CNC(c2nncn2C2CC2)=O)CCC1 C1(CNC(c2[nH]cc(CC)c2)=O)CN(C(=O)CCc2csc(C)n2)CC1C N1(C(C(CC)n2cncn2)=O)CC(NC(=O)CC(C)(C)OC)C2CCCCC12 CC1CCN(C(=O)CCNS(C)(=O)=O)CC1CNC(C1CC(=O)NC(=O)C1)=O c1(C(C)C)cc(C(=O)N(CCO)Cc2ccn(C(C)C)n2)nn1C.C1C(C)C(=O)N1 CC1CC(C(=O)OC(C)(C)C)CCN1Cc1ccc(Br)s1 C1(CNC(c2n(C)ncc2)=O)COC2(COCCN(C(=O)CSC(=N)N)C2)C1 C(=O)(C(CCF)NC(=O)CC(CC)OC)NCC(=O)N(CCC#C)CC N1(C(C2(CC(C)=O)CC2)=O)CC=C(C(=O)NOCCN(C)C)C1 c1(C(=O)NC2CC(C)(NC(c3cn(CCN(C)C)nn3)=O)C2)cccc(CO)n1 C(=O)(C1=CCC2(COC2)OC1)N(CCCN(C(c1cc(CSCC)on1)=O)C)C C(=O)(C1=CC2CCCCCC12)NC(CC(C)NC(C1CC(OCC)C1)=O)C Cc1[nH]c(C#N)cc1C(=O)NC1CCCCC1NC(=O)C(O)C(C)(C)C N1(C(C2C3(CCN(C(C4CC(CC)(CC)C4)=O)C3)C2)=O)CCc2ccncc21 c1(C(=O)O)ccc2c(c1)CN(C(C1CN(Cc3ccncc3Cl)CCC1O)=O)C2 C(=O)(C(C)(C)COCc1ccccc1)NCC1N(C(CC2ON=C(C)C2)=O)CC1 N1(C(CCCCOC)=O)CC(NC(c2ccc(Cl)cc2N)=O)C2(CC2)C1 C1(N(C(C(C2CCCC2)NC(C(C)CN(C)C)=O)=O)C)CC2(CCC2)C1 C1(CN(C)C(c2ccc(CO)cc2)=O)CCCCN1C(C1CSCN1C)=O C1(CC(=O)N(C2CCCN(C(C3CN(C(C)=O)C3)=O)C2)CCC)CCN(C)CC1 C1(NC(=O)NCC2(CC)CCOC2)CCC(NC)CC1 c1(NC(C)=O)ccc(C(=O)O)cc1NC(=O)Cc1nc(SC)ns1 C1(NC(c2c(C)csn2)=O)CN(C(=O)CC2CCCCN2C)CC1N=[N+]=[N-] c1(C(=O)NC(CC=C)CNC(=O)C=CCN(C)CC)ccc(C2CC2)cc1 C1(C(=O)NCC(C(C)C)NC(C2CCCN2C=O)=O)CC(S(C)(=O)=O)C1 Cc1nc2cc(C(=O)NC3(C)CN(C(C4(C)CCCO4)=O)C3)ccc2n1C C1(NC(c2c(CC)occ2)=O)CCCC12CN(C(c1cc(F)n(C)n1)=O)C2 n1(CC)cc(-c2nn[nH]n2)c(O)nc1=O.C12CC(CO1)CNC(=O)C2 C1(C(=O)NCC2CCC(NC(C#CC3(C)CC3)=O)CC2)CCCCC12CCC2 C1(C(=O)NCC=CCC(=O)NCC(C)(O)C2CC2)CCCC12CC2 c1(C(N)=O)ccc(F)c(CN2CCCCC(NC(C3CCS(=O)(=O)CC3)=O)C2)c1 C1(C(N2CCN(CC(C)C)CC2)=O)CC(F)CCN1C(=O)C(C)S(C)(=O)=O C#CCC(CC(=O)NCC1(CO)CCCCC1)NC(=O)C(C)C1CCC1 c1(C(=O)NCCNC2C(CC(=O)N(C)C)CCC2)cccc(OC(F)(F)F)c1 C1(C(=O)NC(CCCCNC(C(CCOC)(C)C)=O)CO)CC2CCCC(C1)C2 N1(C(CSC(C)C)=O)CC(O)(CCNC(C2(Cc3cnn[nH]3)CCC2)=O)C1 C1(C(=O)NC2CC(C)(CNC(c3cn(C4CCC4)nn3)=O)C2)C2CS(=O)(=O)CC12 C1(N(C(C(c2cccc(Cl)c2Cl)C)=O)C)CCCN(C(c2cccnn2)=O)CC1 N1(C(C=C(C)C(F)F)=O)CCC(NC(=O)C(C)(C)C(F)F)C(F)C1 CCC(C)CCOC(=O)C(=O)N(C)CC1CCCOC1 CC(C)CC(O)CC(=O)N(CCC(=O)NCC1(CC2CCC2)CC1)C1CC1 c1(C(=O)OCC2CC(OC)C2)ccc(Cl)c(Cl)c1 c1(OCOC)ccc(C(=O)N(CCC#N)C(C2CCCCO2)C2CC2)cc1 C1(CNC(c2cc(O)nc(O)c2)=O)CC2CCC(C1)N2c1nc(Cl)ncc1F c1(C(=O)NCC2N(C(CC3C(C)(C)COC3)=O)CCOC2)c[nH]nc1S(N)(=O)=O N1(C(c2c(CC)c[nH]n2)=O)CCC(CC(=O)NCC(C2CCOCC2)O)C1(C)C C=CCC(F)(F)C(=O)NCC1CCCC(C(N(C)C[Si](C)(C)C)=O)C1 Cc1cc([N+](=O)[O-])cnc1N1CCOC(c2ccc(OC(F)F)cc2)C1 C12(NC(C(CCCC)C)=O)CCCC1(F)CN(C(=O)C(C)CC(N)=O)C2 C(=O)(C(CO)NC(=O)C(C)C1CC1)N1C(C(C)C)CC1 C1(NC(c2ccc(C(C)C)o2)=O)CCN(C(c2ccc(Cl)cc2N)=O)C1(C)C C1(CC(=O)NCC2CC(NC(CC(C)(C)OC)=O)C(O)C2)CCCC2(CCC2)O1 C1(C(=O)NC2CCN(CCCO)C2)CC2CCC1N2C(c1cnc(O)c(F)c1)=O N1(C(CC=CC)=O)CCN(C(c2ccsc2Br)=O)C(CO)C1 CC1(C)CCCC(C(=O)NCC2(NC(=O)Cc3csc(-c4ccco4)n3)CC2)O1 CCC(C)(C)C(O)C(=O)N1CCC(O)(CNC(=O)CCn2cnnn2)C1 C(c1cnn(C)c1C)=CC(=O)N(CCCNC(C1ON=C(CC)C1)=O)CC C1(NC(C2C(CC)CCCC2)=O)CN(C(=O)CCC=CC(C)C)CC1(C)C CCN=c1[nH]c(C(=O)NC2COCCN(C(=O)CC3CC=CCN3C)C2)cs1 Nc1cccc(C(N2CCCC(NC(c3cccnn3)=O)C2)=O)n1 c1(C(N(C2CCCN(C(c3cnn(C)c3N)=O)C2)C)=O)cnn2c(=O)cc[nH]c12 N1(CC(=O)NC2(C(=O)NC3CCCC(C(C)=O)C3)CCC2)CCS(=O)(=O)CC1 C1(NC(C)=O)CCCC(CNC(=O)C(=O)NCC(F)F)C1 C(C)(CC(=O)NCC1CCN(C(=O)CCC2CC2)CC1)(C(F)F)N(C)C C1(C(=O)NC2CN(C(=O)CC3(O)CC3)CC2O)CCC2(CCC2)CC1 C12(C(=O)NC3CC3)CC1CCN2C(=O)C(C(C)C)C1CCC1.C1(=O)CCN1CC#C c1(NCC(CCC)C)ncc(C)cc1S(=O)(=O)NC(CCO)c1cccs1 N1(C(C(C)CN2CCOCC2)=O)CC(CNC(=O)CNC(N)=O)CC(C)(C)C1 c1(C(=O)NC2(C(C)=O)CCCC2)cc2c(s1)CCN(Cc1ccccc1)C2 C1(NC(CC)=O)CC(CNC(c2ccccc2SCc2nc[nH]n2)=O)C12CCC2 C=C1CC(C(=O)NC(CNC(C2C3COCC23)=O)CC)(C(F)F)C1 Cc1cc(CC(N2CCN(C(N3CCNCC3)=O)CC2)=O)c(C)n1C c1(C(N2CC(N3CCN(C(=O)C#CC4CCC4)CC3)C2)=O)ccn2nccc2c1 N1(C(CC2N(C(C(C)O)=O)CC2)=O)CC([N+](=O)[O-])C1 CC(C)CC(C)(C)C(=O)N1CCC(O)(CNC(C2(O)CCSC2)=O)CC1 c1(CC(=O)NC(C)CNC(C2CCN(c3ccncc3)C2)=O)ccc(Cl)cc1 N1(C(C(C#C)(C)C)=O)CCC(C(=O)NCC2(CC)CCCO2)C(O)C1 c1(CN2CC(NC(C(CCC)C)=O)(CO)C2)ccc(C#N)cc1 C1(C(=O)NCC2=CCN(C(c3cc(C)sc3C)=O)CC2)CCc2n[nH]cc2C1C c1(C(=O)NC2CCN(C(c3c(C)n[nH]c3)=O)C2)cnc2[nH]c(=N)sc2c1 CCC(O)C(F)(F)C(=O)N1CCC1C(N1CC(c2ccncn2)C1)=O C1(OC(C2N(S(CC)(=O)=O)CCC2)=O)CC(=O)N(C(C)C)C1 N1(C(C(C)(C)O)=O)CCC2(C1)CN(C(C1CC3CC(O)CC(C1)C3)=O)CCO2 C12CCN(CC1)C(=O)C1CCOC21.C1(CNC(c2cc(CF)on2)=O)C2COCC12 C1(F)(CNC(CN(C)C(=O)C2CC2)=O)CCCN(C(C2(C)CCCCO2)=O)C1 c1(C(N2CCC(OCCNC(CC(=C)C)=O)C2)=O)cc(S(C)(=O)=O)ccc1C c1(C(N(C(C(=O)NCSc2ccccc2)C2C(CC)C2)C)C)cc2sccc2s1 N1(C(C(C)(O)C2CCOC2)=O)CCC2(CCCN(C(=O)C=Cc3cccs3)C2)C1 c1(C(=O)NCC(CC)NC(=O)CC2CCC(F)(F)CO2)cn2cc(C)sc2n1 C1(C(=O)NC(CCC=C)C2CC2)CNC(=O)CN1C(=O)C(C)OC N1(C(CCC=CCC=C)=O)CC2CN(C(c3c(C)ccc(C)c3N)=O)CC2(C)C1 c1(C(=O)NC(CC(C)C)C)ccc2c(C(N3CC(NC(=O)C4CC4)C3)=O)n[nH]c2c1 c1(OC)ccc(C(N2CC3(CCN3C(C3CN(C(C)C)C3)=O)C2)=O)cc1[N+](=O)[O-] N1(C(CC2(NC(CCNC(N)=O)=O)CCCCC2)=O)CC2C3CCC(C3)C2C1 C1(C(N(C)CC2N(C(CN(CC(=O)NC(C)C)C)=O)CCC2)=O)CC2(C1)CC2F N1(C(c2cccc(-c3nc(C)on3)c2)=O)CCC2(CCCCC2NC(=O)CO)C1 C1(C)(CNC(CN(CCOC)C)=O)CCN(C(=O)C=CC(N2CCOCC2)=O)C1 C(=O)(CC(O)C(C)C)N1CC(C)(OCC(=O)NC2(COC)CCOC2)C1 c1(C(=O)NC(CC)CN(C(=O)COC(F)(F)F)C)ccc(N)c([N+](=O)[O-])c1 N12CC3C(C3C1)C2.n1(CC=C)ccc(C(N2CCCC2)=O)n1 CC(C)CC(C(=O)N(CC(C)O)C1CC1)ONC(c1ccccc1CO)=O CC1(C)OC(=O)CC1C(=O)NC(C(=O)NCc1nc(CO)cs1)C1CC1 C1(OCC)COCCC1CC(=O)NCC(C)CN(C(=O)C(C)SC)C c1(C(N2CC3C(NC(C(CC(C)C)OC)=O)(C3)C2)=O)cn2ccc(C)c(C)c2n1 c1(C(N2C3CN(C(C4(C(C)C)CC4)=O)C(C3)C2)=O)ccc2oc(S)nc2c1 CCC(CC(C)C)C(=O)N1CCN(C(c2n[nH]c(C3CC3)c2Cl)=O)CC1C(C)C C#CC1(O)CN(C(C2CCC2CNC(=O)CN2CCCC2=O)=O)C1 c1(C(C)NC(C(CC(=C)Cl)n2cc(CCOC)nn2)=O)n[nH]c2ccccc12 C(=O)(C(F)CC1CCC1)N1CC(O)C1.C(=O)C(O)C1(NC(=O)OC(C)(C)C)N=N1 c1(C(=O)NC(C)CN(C)C(c2nc(C(C)(C)C)no2)=O)cn2c(n1)CCCC2 C1(OC)CCN(C(c2cccnc2CNC2CC(C(=O)N(C)C)C2)=O)CC1 c1(N2CCN(C3CN(C(C(C)C)=O)C3)CC2)nc2c(cc1C#N)C(=O)CCC2 CCS(=O)(=O)CC(=O)NC1CC1CNC(=O)CCc1ccc(OCC)cc1 c1(CCC(=O)NC2C(NC(c3cnc(C(C)OC)s3)=O)CC2)ccc(Cl)cc1 C(=O)(C1=NOC(c2ccccc2)C1)NCCCN(C(C(C=C)(F)F)=O)CC Cc1cc(C(=O)NC23CC(NC(=O)CN4CCCC4CO)(C2)C3)c2scnc2c1C Cc1nn(C)c(C)c1CC(N1CC(C2(NC(c3ccc(N)cc3F)=O)CC2)C1)=O C1(Sc2ccc(NC(N3CC(N4CCOCC4)C3)=O)cc2)CCCCNC1=O N1(C(=O)C#CC2CCOC2)CCC2(CCN(C(=O)C(O)CC(F)(F)F)C2)C1 c1(C(=O)NCC2C(C)CCN2C(c2cccs2)=O)cc(F)ccc1Cl c1(OC)cc(F)c(NC(=O)NCC2(Cl)CCC2)cc1Cl C(=O)(C#CC1CCOC1)NCC(C(=O)N1CCC(CC(C)(C)C)C1)(C)C Cc1cnc(N2CCN(CC(N3CCOCC3)=O)C(=O)C2)nc1N(C)C CC(C#N)CCC(=O)NC(c1cc(Cl)ccc1Br)C Cc1cccc(CCC(=O)NC(C(C)NC(=O)CCc2cncn2C)C(C)C)c1 C1(CC(=O)Nc2c(OCC)nccn2)CN(C(c2conc2C)=O)C(C)(C)C1 C1(C(N2CCC(NCC3(n4nccn4)CC3)C(C)C2)C)CC2(CCOCC2)C1 N1(C(c2cncc(C)n2)=O)CCCCC(CNC(=O)CC(C)CF)C1 c1(C(C(=O)Nc2ncn(CC)c2)(C)O)ccc(Cl)cc1 c1(C(=O)NC(CNC(c2cc(=NC)[nH]cc2)=O)CO)cc2cc[nH]c(=O)c2s1 N(C(=NCCC(C)C)NCc1csc(C)n1)CC1CCCC(OC)C1 C1(C(=O)NCC2C(NC(CSCCCC)=O)CCCC2)CC2(CCC2OC)C1 C(C)(CC(C)(C)C)(c1n(CCOC)nnn1)NCc1ccc(C#N)s1 O=C1Cc2c(N3CCC(N(c4ncnc5ccccc45)CCO)C3)ncnc2N1 c1(-n2cc(CC(C)C(=O)O)nn2)ccc(C(N2CCCC(F)C2)=O)cc1 N1(CC(=O)NC2CCOC(CNC(=O)C(=Cc3cscn3)F)C2)C(=O)CCC1=O C(C)(C)(C(C)CC(=O)N1CC2(CC(O)C2)C1)NC(Cc1c(C)cnn1C)=O CC(C)C(C)(CNC(C1CCC(C(F)F)O1)=O)NC(=O)C=CC=CC1CCCC1 N1(C(Cc2ccn(C)n2)=O)CCCC(C2CCN(C(c3coc(Br)c3)=O)CC2)C1 CC(CCCCNC(c1cc(C(N)=O)cs1)=O)NC(c1cn(C2CCC2)nn1)=O N1(C(CC(CC)C)=O)CC(C)(C)OCC1CNC(c1ccc2cc[nH]c2n1)=O CC1CC=C(C(=O)NC(CC(F)F)C(=O)NC2(C)CC(C)(C)C2)CC1 c1(CC)ccc(OC(C)C(N2CC3C(N(C(=O)CCF)C)C3C2)=O)cc1 c1(C(=O)NC23C(CN(C(C4C(CCC)C4)=O)C2)C3)cc(Cl)cc2ccc(C)nc12 c1(C(=O)OC)ccc(COC(c2cccc(S(=O)(=O)F)c2)=O)cc1[N+](=O)[O-] CCCC(C(O)C(=O)N(C)CCN1CCCCC1)NC(=O)C1=CCCC1C c1(CC(C)NC(CC)Cc2ccc(Br)cc2)c[nH]c2ccccc12 C1CCC(C2CCCN(Cc3csnc3C3CC3)C2)CC1 C1(C(=O)NCC(CNC(c2cn(C)nn2)=O)(C)O)CCc2ncnn2C1 C=C(F)CN=c1[nH]c2c(c(=NCc3cccc(N(C)C)n3)[nH]1)COC2 C1(NC(CCC)=O)CN(C(c2nnn(CC)c2CC)=O)CC1F c1(CC)nc(CN2CCC2CNC(C2COCCO2)=O)cs1 c1(OCCCNC(=O)CC2CCC2)ccc(OCCO)cc1.C1(=O)CN1.C(CO)O c1(C(C(=O)NC(C)(C)C)N(CCCO)C)ccc(OCC(F)F)cc1 N1(C(c2cc(C)nnc2)=O)CCOC2(CCC(NC(C3CC3C(C)C)=O)CC2)C1 N1(C(=O)CCN2CCCC2)CCCC(C2CN(Cc3cc(Cl)cc(Br)c3O)C2)C1 c1(C(N2C(CCNC(C=NOC)=O)CSCC2)=O)cc(Cl)c(O)cc1C C(=O)(C1=CCCC1C)NC1CCC(CC(=O)NCC)C1 C1(CNC(=O)CONC(c2ncc(Cl)s2)=O)CCCCO1 N1(C(C2C(C(C)C)OCC2)=O)CCC(NC(=O)C=C2CN3CCC2CC3)C(F)C1 n1(CC)cnc2c(N(C)CC3CCN(C)C3)nc(N3CCCC4(CCC4)C3)nc12 c1(C(N2CC(NC(c3ccc(=N)[nH]n3)=O)C(CO)CC2)=O)cnc2ccccn12 CS(C)(=O)=NC(=O)C(=O)NC1(C)CC(NC(c2ccc(Cl)c(Cl)c2)=O)C1 c1cc(C(=O)CBr)ccc1N.C(CCCO)NCC(C)C.C1C(=O)N1C1CC1 N1(C(C(COC)(F)F)=O)CC2(CC(C(=O)Nc3ccc(C)c(CO)c3)CO2)C1 C1(C(=O)NCC(CNC(=O)C(c2ccc(Cl)cc2)N(C)C)OC)CC(=O)NC(=O)N1 C(CC(=O)NC)N(C(=O)C(C)OCC(C)C)CC=C.C1(N(C)C)C(=O)N2CC1C2 C(=O)(C(O)CC(F)(F)F)N1C(C(N(C)Cc2ncccn2)=O)CCCC1 N1(C(CC(C)OC)=O)CCC2(CC1)CCN(C(C1(Cl)CC1)=O)CC2C C#Cc1ccc(C(=O)NCC=CCNC(c2c(Cl)nn(C)c2C)=O)cc1Cl N1(C(CCS(C)=O)=O)CC2CCN(C(=O)C(F)C(C)(C)O)CC12 Cc1cn2ccnc(C(N3CCCC3CNC(C3CCC(=O)O3)=O)=O)c2n1 N1(C(CCCOCC)=O)CCC(C)C1C(=O)N(CCC(C)C)C c1(CC)nc(C)oc1C(=O)NCC1(C)CCCN1C(C1CN(C)CCO1)=O CCCC(CCNC(C1CC(NC(c2cc(O)nn2C)=O)CCO1)=O)C1CC1 N1(C(C(C)C)=O)CCC2(CCCC2NC(c2cc(CF)on2)=O)CC1 C1(C(=O)NCC2(O)CC(CNC(=O)C3=CCOCC3)C2)CCS(=O)(=O)C12CCC2 N1(Cc2cnn3ccnc(C)c32)CC2(CN(C(=O)OC(C)(C)C)CC(C)(C)O2)C1 c1(CC)c(C(N2CC(C)(C)CC2CNC(=O)C(C(C)C)NC=O)=O)cccc1C N#Cc1c(Cl)nsc1N1CC2CC(NC(C3CCC(=O)N3)=O)C2C1 C1(C(=O)OC)CC12CCN(C(=O)N(c1ncc(Br)s1)c1ccccn1)CC2 C12(C(N3CCCC(N(C(=O)CC4(CO)CC4)C)C3)=O)C3C4C1C1C2C3C41C c1(C(=O)NCCC2N(C(C(CC)N(C)C)=O)CCC2)cnc(O)cc1O C(=O)(C1Cc2c(Cl)cccc21)N1CC(OC)(CNC(C2(C)CCC(C)C2)=O)C1 c1(OC)cccc(C)c1C(=O)NC(C1CCCCN1C(=O)C=Cc1cc[nH]n1)C C1(NC(=O)CCCc2cnn[nH]2)CN(C(=O)C(F)F)CC2(CC2)C1 C#Cc1cc(C(=O)NC(C)CCN(C)C(c2cnn(C3CCC3)c2)=O)cc(F)c1 c1(C(=O)NCCC(CNC(C(C)SCCCC)=O)O)ccc2cccnn12 c1(C(N2CC(OCCNC(=O)CC3CC3(Cl)Cl)C2)=O)ccc2nnc(S)n2c1 C(CCC(N)=O)(C(=O)NC(C)(C)CCNC(c1cnnc(O)c1)=O)N(C)C Cc1ccc(C(=O)NC(c2ccccc2)C(C)NC(C2C(C)(C)C2(C)C)=O)nn1 C1(C(=O)NCC(C)(C(C)C)NC(C2(OC)CC2)=O)CC2(C1)CC21CC1 C#Cc1cccc(CNC(CCCC=C)C(=O)NCCC(=O)OC(C)(C)C)c1F CC(CCCCNC(=O)C(C1CCCCC1)O)NC(=O)C(=O)NOC C1(NC(c2ccc(F)cc2)=O)CC2CN(C(C3CCN(C4CC4)C3)=O)CC2C1 c1(C(=O)NCC2CC(O)(CNC(CNC(=O)OC)=O)C2)ccc(C#N)cc1O c1(C(=O)NC2C(C)CCNC2=O)c2c(nn1C)CCSC2 C1(O)(C(N2CCCC(C(=O)NCC(COC(C)C)O)C2)=O)CCCCCC1 c1(C(c2n(CCC)nnn2)NCC(CC(C)C)OC)ccc2nc[nH]c2c1 S(=O)(=O)(c1ccccc1CCl)Nc1c(OC)cc(C)c(C)c1 C1(NC(COCC(=C)C)=O)CCC(C)N(C(c2cc(-c3ccco3)[nH]n2)=O)C1 c1(C(C)NC(C(C2CCCO2)NC(C(=Cc2cn[nH]c2)C)=O)=O)cccnc1O C(=O)(C(C)(C)CNC(C)=O)N(CC=CC(=O)NC(COC)C(C)C)C c1(C(=O)NCC(CNC(C2(C3CCCO3)CCC2)=O)OC)c(Cl)n[nH]c1C C1(c2nnnn2CCC23CC(CO2)C3)(NCCn2ccnn2)CCCC1 N#CC(CCc1ccccc1)C(=O)NCC1CN(C(C2(O)CCOC2)=O)CCO1 N1(C(CC2ON=C(C)C2)=O)CCC(NC(C2(C(C)C)CCC2)=O)C(F)C1 N1(C(C2CC(C(C)C)C2)=O)CCC(=CCNC(=O)C(F)(F)C2(O)CCCC2)CC1 C1(C(=O)NC2C(NC(C3ON=C(C)C3)=O)CCC2)CC(=O)NC(=O)C1 N1(C(c2cccc(C)c2O)=O)CCN(C(C2(C)CC=CC2)=O)CC(C)(F)C1 CCCCCCN(CCCCCC)C(C(C)(C)CO)C1CNC1 c1(C(=O)NCC2(CNC(C(CC)SC)=O)CC23CCC3)cccc2[nH]cc(Cl)c12 C=CC(C)(C)CC(=O)NCCC(C)NC(=O)Cc1ccccc1CC#N c1(C(=O)NC2C(NC(c3cc(O)cs3)=O)CCCC2)cc2n(n1)CCO2 c1(C(=O)NC(CNC(CCC(C)OCC)=O)(C)CO)cc(O)ccc1F CC1(C)CCOC(CC(N2CC(NC(c3ccc(F)c(Cl)c3)=O)C(O)C2)=O)C1 C1(C(=O)NC2C(CNC(C(C)C3CCOC3)=O)CCCC2)C(F)(F)C12CCC2 c1(C(N(CCCN(C(=O)CCC2CCCO2)C)C)=O)cc2nc(F)ccc2o1 N1(C(=O)NC(c2ccc(C#N)cc2)C(C)C)CC2(CC2)c2ccc(Br)cc21 N1(C(C(C=C=C)C)=O)CC(NC(c2ccn3nccc3c2)=O)CC2(CC2)C1 C1(NC(COC(C)C)=O)CC2CN(C(=O)CCc3ccccc3F)CC2C1 C1(O)(CCNC(C2CC3CCC3C2)=O)CCN(C(C2COC(=O)C2)=O)CC1 S(=O)(=O)(c1ccc(Cl)cc1)NC(C(=O)Oc1cc(C(=O)NCC)n(C)n1)C(C)O N1(C(CCc2c(C)noc2Cl)=O)CCN(C(=O)CC(F)F)C2(CCC2)C1 C1(C(C)CO)CCN(C(=O)CCOCCN(C(=O)C(C)n2ccnc2)C)CC1 C(=O)(C(CNC(=O)CC1CCOC1(C)C)C(C)(C)C)N(CC(CC)O)C c1(C(=O)NC2CCCC(NC(C(C)=CC3CC3)=O)C2)c(C)cncc1C c1(CC(=O)NC2CCCN(C(CC=CC=C)=O)C2C)coc2ccc(F)cc12 c1(C(C)OCC(=O)N(C)CCNC(C2CCCN2C)=O)nccn1C n1(CC)cc(Cl)c(C(=O)NCCC(C)NC(=O)CNC(c2ccc(O)cc2)=O)n1 C(=O)(C1CCCc2n[nH]cc21)NC1C2CN(C(C=Cc3c(C)ncs3)=O)CC1C2 N1(C(C(F)=C(C)C)=O)CCN(C(c2cnc(C3CCC3)cc2C)=O)C(CO)C1 C1(O)(c2ccc(C)cc2)CCN(S(=O)(=O)N2CCCCc3ccccc32)CC1 N1(C(C2N(C(CNC(=O)OC)=O)C(C)CC2)=O)CCCC(N=[N+]=[N-])C1 C1(=CC(N2CCC(NC(=O)CC3CC=CC3)C2)=O)C2CC3CC(C2)CC1C3 C(=O)(C(CC(F)F)N(C)C)NC(c1cc(C(F)(F)F)ccn1)C C1(C(N(C2CCN(C(=O)CCc3cc[nH]n3)CC2)C)=O)CC2C=CCC(C1)C2 C(C)(C(C)(C)CO)NC(CC1C(NC(CC2ON=C(C)C2)=O)CC1O)=O CN1CCC2(CN(C(=O)NCc3c[nH]nc3C(F)F)CCO2)C1 C1(C)(CCNC(C2CC(SC)C2)=O)CCN(C(=O)Cc2cccn2C)C1 CCC(CCC(=O)NCCN(C(=O)Cc1cnn(C2CC2)c1)CC)OC c1(OC)ccc(Cl)c(CC(N2CCCC(N3CCCCC3=O)C2)=O)c1F C1(c2ccc(F)cc2)(NC(=O)NCCCc2cccs2)CCCCC1 c1(C(C)=O)ccccc1NC(=O)Cn1cc(C2(N(C)C)CCOCC2)nn1 C1(NC(=O)COC2CCCC2)COC2(CCN(C(c3cc(F)cs3)=O)C2)C1 C1(C(=O)NCCCSn2cc(CNC(=O)OC(C)(C)C)nn2)CCN(C(C)=O)C1 C=C1CCC(C(=O)NC(C2CCN(C(=O)CCC3CC(F)(F)C3)C2)C)CC1 c1(C(=O)NCC2CC(NC(c3c(NC)nccc3)=O)C2)c(F)ccc2n[nH]cc12 N1(C(CCCC#C)=O)CCC2(CCCN2C(=O)C(CC(F)F)c2ccccc2)C1 C1(C)(CNC(c2ncc(CC)cn2)=O)CCN(C(c2ccc(C3CC3)s2)=O)CC1 c1(CC)cccc(NC(C2CN(C(=O)CC3C=CCC3)CC2C(C)C)=O)c1 n1(CC(N2C(COC)CN(C(C3(N=[N+]=[N-])CC3)=O)CC2)=O)nnc2c1CCCC2 C1(NC(Cn2ncc(C)c2)=O)COCCN(C(C2(CF)CCC2)=O)C1 Cc1c(C(N2CCCC(F)(CNC(C3(O)CCC3)=O)C2)=O)oc2c1C(=O)CCC2 c1(C(=O)NC2C(NC(Cc3cc(C)sc3C)=O)C2)c[nH]c2ncccc12 N1(C(C2CCCC3(CC3)C2)=O)CC2CCCC(C1)N2C(=O)C=Cc1ccco1 N1(CC(C)C)N=C(C(=O)NC2(CO)CCCN(C(=O)CC(C)SC)C2)CCC1=O C1(CNC(c2ccc(C3CC3)cc2)=O)CN(C(C2CCC(F)(F)C2)=O)CC12CC2 C(=O)(C(F)C(F)(F)F)NCCCN(C(c1[nH]cc(C(=O)OC)c1)=O)C c1(CN2CCC(C(C)NC(c3scc(C)c3)=O)CC2)ccc(C)cc1Br c1(C(=O)OCC)nc(C(C)NCC2CCN(C(=O)OC(C)(C)C)CC2)oc1C C#CCC(C(=O)NCCC(O)COC)NC(c1nnc(S)n1C)=O c1(C(c2n(CCCCCC)nnn2)NC2(CCO)CCCC2)ncc(C)cc1Cl c1(NC(CCSCC(C)C)=O)ccccc1Sc1ccc(Cl)s1 C(=O)(C(C)(C)S(C)(=O)=O)NCCC1N(C(c2[nH]cc(OC)c(=O)c2)=O)CCSC1 CC1Oc2ccccc2OC1C(=O)NC1C=CCN(C(=O)C2=C(Cl)CCCC2)C1 Cc1c(C(=O)NCCCCN(C)C(c2ncc[nH]c2=O)=O)[nH]ccc1=O C1(NC(c2c(C)nc(C)o2)=O)CN(C(=O)CC2COCC2(C)C)C2(CCC2)C1 N1(C(CC(C)C)=O)CCC2CCC(C1)N2C(=O)Cc1ccc2c(n1)NCCC2 CCCCC(=O)NC1CC(NC(C2(CCF)CC2)=O)C1 c1(Cc2nnc(N3C(CC)C(C)CC3)n2C2CC2)cc(C)c(OC(F)F)c(C)c1 N1(C(C2CCC(=O)O2)=O)CC2(CC2)CC1CNC(c1csc(Cl)c1)=O N1(C(C(CSC)OC)=O)CC2CCCC(C1)N2C(c1cccc2ncccc12)=O CCC(C)C(O)C(C)C(=O)NC1CCOC1C(N1CC(C)C(F)(F)C1)=O C1(CNC(C2CC(C)(C)OCC2)=O)C2CCCC1N(C(=O)C1=NNC(=O)C1)C2 c1(C(N2CCN(C(CC(C)OC)=O)C(C(F)F)C2)=O)cnc2ccnn2c1 c1(NC(C2C(C(N3CCCC(C#N)C3)=O)C2)=O)ccc2nnsc2c1 Cn1[nH]c(CN)nc1=NC(=O)C(Cc1ccccc1)C(F)(F)F c1(C(N2C(CNC(c3c(C)nc[nH]3)=O)C3CCC2C3)=O)noc2c1CCCC2 N1(C(CNC(=O)OC)=O)CCN(C(C2CCCC2c2nncn2C)=O)C(C2CC2)C1 C1(C(=O)NC2C(CNC(C(CC)N3CCCC3=O)=O)C2)CN(C)CC1C(F)(F)F c1(C(=O)NCC2N(C(C3OCCN(C(C)=O)C3)=O)CCC2)cnn2ccccc12 N1(C(C2C(C)(CC)C2)=O)CC=CC(NC(c2cnc(OC)cn2)=O)C1 CC(C)CC(C(=O)Nc1cnn(C(C)C)c1)NC(=O)C(C)O N1(C(C2C(=C)C2)=O)CCN(C(c2cnc(Cl)c(N)c2)=O)C(CC(F)F)C1 C1(NC(CC(CC)OC)=O)CN(C(=O)CCc2cccc(C#N)c2)C2CCCC12 N1(C(c2cnn(CCC(F)(F)F)c2)=O)CC2(CCCC2NC(C2(O)CCC2)=O)C1 N1(CC(COCCOC)O)CC(C)(C)CCC1CNC(c1cc(C)no1)=O c1(C(=O)OC)cc(N(C(C)CNC(c2conc2C(F)(F)F)=O)C)ncn1 c1(C(N2C(CNC(C34CC(C)(C3)C4)=O)CCC2)=O)ccc(S(N)(=O)=O)c(Cl)c1 N1(C(C(C)N(C2CCN(C)C2)C(C2(C)CC=CCC2)=O)=O)CCOC2(CCC2)C1 c1(CNC(CCOC2CCN(C)CC2)=O)nn(C)c2c1CN(C(=O)CCF)CC2 CC(C(=O)NC(C1(O)CN(C(=O)CNC(c2ccoc2)=O)C1)C)C(F)(F)C(F)F CC(C)(O)C#CC(=O)N1CCC(CCC(=O)N(CCCO)C2CC2)C1 C(=O)(C(C)S(=O)(=O)C(C)C)NC1CN(C(c2cn(CCC)nn2)=O)CC(O)C1 c1(NC(C2C=CC(=O)N=N2)=O)c(-c2ccc(C(F)(F)F)s2)ccc2c1OCO2 c1(N(C)C)cnc(C(=O)NCCC2(NC(=O)CC3COC(=O)C3)CCCC2)cn1 N1(C(CC(CC)C2CCC2)=O)CCOCCC1C(=O)NCC1CN(C(=O)OC)C1 C1(NC(=O)NCC2C(C(=O)OC)CCO2)CCCN(CCCO)C1 CCCCC(CNC(=O)C=Cc1cccs1)NC(=O)Cn1ccc(C(F)F)n1 c1(C(=O)NCC2(CNC(c3cnnn3C3CC3)=O)CC2)ccc(-n2ccnn2)cc1 N1(C(=O)CCc2nncs2)CCN(C(c2cc(O)nc(C3CC3)n2)=O)CC(O)C1 C#CCCCCCC(=O)N1CCC(NC(=O)C=CCOC)C12CCC2 Cn1cccc1C=CC(=O)NC1CCCCC1NC(c1cscn1)=O c1(C(CO)NC(C)C(=O)Nc2ccsc2)c(F)cccc1F N1(C(C(CC)C#N)=O)CC(C)CN(C(c2cccc3nc(CO)[nH]c23)=O)C(C)C1 C12(NC(C3CCN(C(c4ccnc(O)c4)=O)CC3)=O)CCC(CC1O)C2 C1(C)(NC(C=CC(C)(C)SC)=O)CCN(NC(=O)CSC(F)F)C1 N1(C(C(C=C)(F)F)=O)CCCC(CCNC(C2CCCCC2O)=O)CC1 CC1(C)CC(CNC(C2CCN2C2CCCC2)=O)CN1C(=O)C1=CCCCO1 CCC(CC(=O)N1CCCC(C)(NC(=O)CCOCC(F)(F)F)C1)C(F)F C(=O)(C(O)CC(C)(C)C)NCC1(NC(C2N(C(C)=O)CCC2)=O)CC1 N1(C(c2cn(C(C)C)c(=O)cc2)=O)CC=C(CCNC(C2CCC(=O)N2)=O)CC1 N1(C(CCC=CC(C)C)=O)CC2CCOC2(CNC(=O)Cc2cncnc2O)C1 CCC(C)(CNC(=O)CCCC(C)NC(=O)CC1CCC(=O)N1C)C(N)=O C12(NC(C=CCC)=O)CCC(CN(C(=O)C(C)OCc3ccc(C)cc3)C1)C2 CCCCC(F)(F)C(=O)N1CC2(CCC2)CC1CNC(=O)C(=O)NOC c1(C(N(CCC(=O)NCC#CCOC)CCO)=O)ccc(C#N)[nH]1 C(c1cnccc1C)=CC(=O)NC(CN(C(C(C1CCCC1)OC)=O)C)C CC(C)C(F)(CNC(=O)CCC1CCCCO1)C(=O)NCc1cn(C)cn1 C1(C)(CC)CCNC(=O)CC(=O)N1.C=CCNC(C)=O CCC(C)C(C(=O)NC(C)CCSC)NC(=O)C=CCN(C)C CS(=O)c1ccc(CC(=O)NC2(NC(=O)C(C)(O)C(C)(C)C)CC2)cc1 c1(C(=O)NCC2CC(NC(c3c(C)oc(C4CC4)n3)=O)C2)cc(Cl)nnc1O N1(C(C(CCC2CC2)NC(C(C)n2cnnn2)=O)=O)CCOC2(CCC2)C1 C(CCC(C)CC(=O)NC1CC(C)N(C(C23COC(CCO2)C3)=O)C1)=C(C)C c1(C(C)O)ccc(C(=O)N(C2CSC2)C)cc1.c1(C)cn(C2(C=O)CC2)nn1 N1(C(C2(OC)CS(=O)(=O)C2)=O)CC2CCC(CNC(c3cc[nH]n3)=O)C2C1 CC1(C)CC(NC(=O)CCCNS(C)(=O)=O)CN(C(c2ccc(=N)[nH]c2)=O)C1 C(=O)(C(C)(C)CC(F)F)N1C(C(N2CC=C(COC)CC2)=O)CSC1 c1(C(=O)NC2CCC(O)C2)cn2c(n1)C(C(=O)NC(C)(C)CNS(C)(=O)=O)CCC2 c1(CC(c2nnnn2C)NCCC(C2CCCC2)OCC)ccccc1C Cc1nc(NCC(CO)C(F)(F)F)cc(N(C)Cc2nnc(C(C)(C)C)s2)n1 C(=O)(CC(C)C(F)(F)F)NCC(CC)(C)C(=O)NC(C)CNC(=O)OC c1(C(C=C)O)cn(CCCCCNC(=O)Cc2ccn(CCCCC)n2)nn1 N1(C(c2cc(C)cc(O)c2)=O)CC2CCC(NC(=O)C=C3CCN(C)C3)CC2C1 CC1(C)C2CCC1(C)C2C(=O)NCCCCNC(c1cc(C2CC2)[nH]n1)=O c1(C(=O)NC2C(NC(C=C(C)c3ccco3)=O)CCC2)cc(C)cc(Cl)c1 c1(OC)cccc(Cl)c1C(=O)N(C)CCNC(C1(c2cnn(C)c2)CCCO1)=O n1(COC)cc(NC(c2ccc(C3CCC34CCC4)cc2)=O)ccc1=O CC1CC(NC(c2cc(Cl)c(Br)s2)=O)CN1C(c1cncn1C)=O S(=O)(=O)(c1ccc(C(=O)NCC2CC(O)CN2C(c2cc(OC)cs2)=O)o1)NC c1(C(=O)NC2CCN(C(Cc3cccc(CC)c3)=O)C2)cc2oc(Br)cc2[nH]1 c1(C(=O)NCC2N(C(CC(C(C)C)C)=O)CCCC2)ccc(C#N)c(F)c1 C1(NC(C(C)(C)OC(C)=O)=O)CCCCC1NC(=O)CCCc1nccs1 c1(CNC(C2CC(C(N(C)C)=O)C2)=O)ccc2oc(O)nc2c1 CCC(CC)CCC(=O)NCCCC1CN(C(=O)CSCC(C)C)CCO1 C(=O)(CS(=O)(=O)C1CC1)NCCC1(CNC(Cc2c(Cl)cn(C)n2)=O)CC1 C12(C(N3CCC(NC(=O)OC)C3)=O)CCCC1CCN2C(c1cnc(C)c(C)c1)=O N1(C(C(C)OC)=O)CC(n2cc(Cc3ccc(NC(C)C)cc3)nn2)C(C)C1 C(C)(C(=O)N1CCCCO1)(N(C(CCc1cc(C)[nH]n1)=O)C)C1CC1 C1(NC(COCC(C)C)=O)CC(C(=O)N(C2CC2)CC2(C)CCC2)C12CCC2 c1(C(=O)NC2CCC(NC(C=C(C)C3CC3)=O)C2)cc2c(Cl)cc(Cl)cc2[nH]1 C(CCC(O)C(=O)N1CC(CO)C1)NC(c1c(OC)nccn1)=O CC1(C(=O)N2CCC3(CC2)CC3CNC(=O)C2=C(Cl)CC2)CCc2ccccc21 C1(C2CCCN(C(=O)CCNC3CC3)C2)(NC(C(c2c(C)nn(C)c2)C)=O)CC1 C(=O)(C(C)C1OCCc2ccccc21)N1CCC(c2ccccc2)(COC(C)=O)C1 N1(C(CSC(C)C)=O)CC(CNC(=O)C(=O)NC(C)C)CC1C C1(NC(CCCN(C)C)=O)CC2CC(NC(=O)COCC3CCCCO3)CC12 C1(CNC(C(CCC)=CCC)=O)CN(C(=O)C(C(C)C)SC)CC12CCOCC2 C1(F)(C(=O)NC2CCN(CCOC)C2)CCN(C(C2CCC(=O)NC2)=O)C1 c1(NC(c2c(CC)nc(C)s2)=O)ccc(F)nc1CN1CCC(CC(=O)NC)C1 C(CC(C)(C)C(=O)NCCc1nccs1)NC(CCC)=O C=CCC(C(=O)N1CCC1C(N1CC(O)C1)=O)NC(C)=O Cc1cc(O)nnc1C(N1CCCCC1CN(C(=O)CCCN=[N+]=[N-])C)=O N1(C(c2c(C)ocn2)=O)CC(CCNC(c2ncccc2C(F)F)=O)OC(C)C1 C1(C(=O)NC2CCN(C(C(c3ccc(C)cn3)(F)F)=O)C2C)COCC(C)(C)O1 Cc1cnc(CCC(N2CCCC2CNC(=O)C(C)(C)NC(=O)C(F)(F)F)=O)[nH]1 N1(C(CCOCC)=O)CCC(=CC(N2CC3CC3C2)=O)CC1 c1(NC(C2C(C(=O)NCC(C)(C)C)C2)=O)cc(Cl)c(Br)c(Cl)c1 N1(C(C(CCC=C)NC(c2[nH]nnc2CC)=O)=O)CC(=O)NC(=O)C1C N1(C(C=C(C)C(F)F)=O)CCC(CC(=O)NCc2nc(C)co2)C1 c1(NC(=O)NCc2cc(Oc3ccccc3)ccn2)coc2c1C(O)CCC2 C(=O)(C#CC1CCOC1)NC1C(C(=O)NC2C(C#C)CCC2)COC1 c1(C(=O)NC(C(C)NC(c2c(CC)noc2)=O)CO)cccc2nc(O)n(C)c12 c1(C(=O)NC2CN(C(C(=O)NCC3CC3)=O)C2)cncc2ccccc12 C(c1cccc(Cl)c1)=C(C)C(N1C2CCC1C(NC(C1COC(=O)N1)=O)C2)=O Cc1cc(CN2CC3CC3(C(=O)N=c3nc[nH]s3)C2)cnc1Cl C1(NC(c2cccn(C(C)(C)C)c2=O)=O)CC2CC1CN2C(c1cc(Cl)no1)=O Cc1ccc(CCC(=O)NC(C)CN(C(=O)CCCC(C)O)C)c(C)c1 CCCCC(CC(=O)N1CCC(O)C(O)C1)NC(=O)CCC(C)CC C(C)(C(=O)N=c1ccn(C)[nH]1)N(CCC)C(c1cc(C(C)=O)on1)=O CC(C)(CC(F)F)C(=O)NC1CCC(C)(CNC(C2C=CCS2)=O)C1 Cc1cc(=NCc2nnc(C)n2C)[nH]c(=NCC2(c3ccc(Cl)cc3F)CC2)[nH]1 N1(C(C=NOC)=O)CC=C(CNC(C2CCCC(OC(F)(F)F)C2)=O)CC1 CC1(C)CC(CO)(NC(=O)CC2(C#N)CCOCC2)CO1 C1(F)(C(=O)NC(COCC)CO)CCCN(C(=O)C(C)NC(=O)OC)C1 CC1C=C(C(=O)N(C)CCC2CCN(C(c3cncc(F)c3)=O)CC2)CC1 N1(CC)CC(CNC(=O)CCC2CCCCN2C(=O)CNC(C)=O)OC1=O C(C(C)(CC)C(=O)N=c1cc(COC)n(C)[nH]1)Oc1c(OCC)cccc1 c1(OCCC)ccc(C(=O)NCC2CCCN(C(c3cnc(C)cn3)=O)C2)cc1 c1(C(C(=O)NC)N(C2CC2)Cc2cnn(CC)c2)ccc(O)c(OC)c1 C1(OCC)CC2(C1)CC2C(N1CCC(N(C)C(c2cccnc2NCC)=O)C1)=O N1(C(c2cc(CC)on2)=O)CC2COCCC2(NC(=O)CC2CCCCC2)C1 C(=O)(C1=CCC(F)(F)CC1)NCCCCCNC(c1c(OC)ccc(O)c1)=O C1(CNC(C2C(C(C)C)C2)=O)CCCCN(C(=O)CSc2nccn2C)CC1 Cc1ccc(C(F)(F)C(=O)NCC2(CNC(C3CC3Cl)=O)CCC2)cc1 CC1(C)CC1(C)C(=O)NCCc1cc(C(=O)NCC(N2CCCC2)=O)no1 Cc1ccc2cc(C(N3CCN(C(=O)CCn4cnnn4)C4CC34)=O)ccc2c1 CC(C)CC(C)(O)C(=O)NCc1nc(C(=O)NC2CC(=O)N2)co1 C1(C(=O)NC2CCCC2CF)Cc2c[nH]cc2S1(=O)=O c1(C(=O)NCC2(C)CCCN(C(C3CC(F)(F)C3)=O)C2)ncnc2c1CCCC2 Cc1cc(C2CC2C(N2CC(O)(C#CBr)C2)=O)cc(F)c1 CC(C)CCCCNCC(N1CCN(C)CC1)C1CCCC1 C(=O)(C(CNC(=O)C(C)NC=O)CC(C)C)NC(CCC)CO N=c1nc(CCC(N2CCC(C(=O)Nc3cnn(CCO)c3)C2)=O)[nH][nH]1 Cc1cccc(OCC(=O)NC(CNC(c2ccc(Cl)cc2F)=O)C2CC2)c1C CC1(C)COCCC1C(N1CCC(CO)(CNC(C2CCC3CC2CO3)=O)C1)=O c1(CN2C(C(N(CC#N)CC#N)=O)C3CCC2C3)c(Cl)[nH]c2ccccc12 Cc1cc(NC(C2CC(O)(CNC(=O)CC3CCOC3C)C2)=O)ccc1F C1(NC(C(C)=C2CC2)=O)CN(C(=O)Cc2nccn2C)C2CC12 C1(C(N2CC(N(C(CCOC(C)C)=O)C)C(F)C2)=O)Cc2n[nH]cc2C(=O)N1 Cc1ccc2snc(NC(C)C(C)CCCC(C)C)c2c1 N1(C(=O)COC(F)F)CCOC2(CCS(=O)(=NC(=O)c3coc(Br)n3)CC2)C1 Cn1nnc2c1CCC(C(=O)NCCCCCNC(=O)CC1COCC1O)C2 n1(CC(=C)C)nnnc1C(CCC1OCCO1)C1(CCC(F)(F)F)CC1.N C1(C(N2CC(CNC(CCSCCC)=O)(COC)C2)=O)C(Cl)(Cl)C12CC2 N1(C(C2=CC(C)(C)C2)=O)CC2CC1CCN2C(C1CC(C)(C)C1)=O CC1CN(C(c2cn3ccccc3n2)=O)CC(C)N1C(c1ccc([N+](=O)[O-])[nH]1)=O N1(C(c2cn(CCC)nc2C)=O)CC2CC1CN(C(=O)CCS(N)(=O)=O)C2 c1(C(N2C(C(=O)Nc3ccn(CC)n3)CC(F)(F)C2)=O)cc2ccc(Cl)cc2s1 c1(C(N(C2CCCCC2NC(C2CC=CC2)=O)C)=O)c(F)cc(Br)cc1F C1(CCNC(c2cnn(C3CCCC3)c2)=O)CCC(NC(C2CS(=O)(=O)C2)=O)C1 C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC1C(CC)CN(C(C2C3CCCC23)=O)CC1 c1(C(=O)NC(C(C)NC(=O)C(F)(F)C(F)F)(C)C)cc2ccc(Cl)cc2[nH]1 C(=O)(C(C)(C)C(C)(C)O)NCC1(NC(C(c2cc(F)cc(F)c2)C)=O)CCC1 CC1CSCCCN1C(c1nc(F)ccc1Br)C(=O)NCc1cccc(Br)c1 c1(C(=O)NCC2CCCN(C(C(CCC)OC)=O)CC2)c(Cl)ccc(F)c1C S(=O)(=O)(c1ccc(C(=O)NCC(C2CC2)NC(=O)CC2CC2)cc1)NC(C)C CCC(C)(C)C(=O)C(=O)NCC1CN(C(C2CC2C)=O)CC1C(F)(F)F CC(C)C(C)C(C(=O)O)NC(c1cc(=O)c(Br)c[nH]1)=O Cc1c(O)ccc(C(N2CCCC2c2cn(Cc3cnn[nH]3)nn2)=O)c1C C(CC1=CCN(C(C2CCc3nn[nH]c3C2)=O)CC1)NC(C)=O CCCCC(C(=O)NCC1CCC1CO)NC(=O)CC(C)(C)COC O=C(CS(=O)(=O)c1ccccc1F)N(C1CC1)Cc1cn(-c2ccc(F)nc2)nn1 C1(NC(CCC)=O)CCN(C(=O)C(C(C)C)OCC)CC1C n1(C2C(SC)C2)c(-c2ccc3c(c2)CCC3)csc1=Nc1cccc(C(N)=O)c1 C1(CNC(CCC=C)=O)CN(C(c2ncccc2O)=O)C2CC12 C1(CC=C)(NC(c2nccs2)=O)CCCN(C(C2CCCCC2)=O)C1 CS(=O)(=O)C(C(=O)NCC1(CNC(C2CCC(C)CC2)=O)CC12CCC2)C1CC1 N1(C(C)C(=O)NCc2ccc(C(=O)NC3C(C)(C)C3(C)C)cc2)C(=O)CCC1=O N1(C(C2CCN(C(C3CC(C(=O)OC)C3)=O)CC2)=O)CC(C(C)C)CCC1C n1(CCCC)ncc(C(=O)N(CC(C)(C)CNC(C2CCC2CF)=O)C)c1C Cc1cnc(C(=O)NC2CCCN(C(=O)CC3(O)CCCCCC3)C2)cc1C C(=O)(C(CNC(c1cc(C)c(C)s1)=O)CC1CC1)NC(C#C)(C)C1CC1 Cc1cc(Br)cc(C)c1N1CCC(NC2(c3nnnn3C)CCN(C)C2)C1=O n1(CCC(=O)NCC2(CNC(C3(C)CSC3)=O)CCC2)ccc2cc(Cl)ccc12 C1(C(=O)NC2CCC2C(N2CCC2CC2CC2)=O)CC2C=CC1C2 C(=O)(C1=NOC(C)(C)C1)N1CCC(CC(N)=O)(NC(c2n(CC)nnc2)=O)CC1 c1(CCNC(COCCC)=O)ccc(CNC(c2ccc(C)o2)=O)cc1 c1(C(=O)NCC(CO)NC(c2c(OCC)ccs2)=O)cnc2c[nH]nc2c1 Cc1cc(S(=O)(=O)NC2(C3CCOC3)CC2)c(C)c(S(C)(=O)=O)c1 C1(CNC(C=C(C)c2ccco2)=O)CC(F)(F)CN1C(c1cc(C)on1)=O C(=O)(C(CO)C(C)(C)C)NCC(CC(=O)N(C(C)C(=O)OC)CC)C C(=O)(C(C(C)(C)C)NC(N)=O)N1CC(F)(CNC(C=C(CC)CC)=O)C1 C1(O)(C(C(=O)NCC(CC)N(C(C=C(CC)CC)=O)C)F)CCCC1 C1(C(N(CC(O)C(C)(C)C)C)=O)CCN(C(c2cccc(F)c2)=O)C(C)(C)C1 N1(C(C(C)NS(C)(=O)=O)=O)CCC2(CCC2)C(NC(=O)COCc2ncnn2C)C1 C=CC(C)(CCOC)C(=O)NCCCN1CCN(C(=O)C=CC2CCCO2)CC1 N1(C(c2ccc(C)c(F)c2)=O)CCCC2C1CCCCN2C(=O)C(O)CC(C)C C1(COC(C)C(=O)NC23CC(CNC(C4CCC(=O)N4)=O)(C2)C3)CCCCO1 Cc1ccc(F)c(C(=O)NCC2CCN2C(=O)C(F)(F)Sc2cnn(C)c2)c1F C1(CNC(CC(=C)C)=O)CC2(CCN(C(=O)CCc3cnn(C)n3)C2)CO1 CC(c1cccs1)=CC(=O)NCCCC(C)NC(=O)C(C)(C)C1CCOC1 Cc1cccc(C)c1NC(=O)C(c1cn[nH]c1)N(CCC(C)C)C1CC1 c1(C(=O)NCC2N(C(C(CC)O)=O)CCC2)cc(C)nc2c1cnn2CC C(=O)(C(O)CC[S+](C)C)NC(CNC(CCCC#CC)=O)C1CCC1 N1(C(CCCNC(C=CC(CC)C)=O)=O)CC2C(C(=O)NC)C2C1 CC1COC2(CCC2)CN1C(=O)CC1CN(C(=O)COC2CC2)CC12CC2 Cc1cccc(C)c1C(=O)NCC1(CC(=O)NC(C)C(C)F)CC1 CCC(C)(C)C(C)CC(=O)NC12CC(NC(=O)CSC3CC3)(C1)C2 C(CCN=C(NC(C)C)N1CCN(Cc2ccc3c(c2)OCO3)C(=O)C1)OC c1(C(=O)NC2C(NC(C(C)OC)=O)CCCC2)ccc2c(c1)CCO2 CSC1=C(C(=O)N(C2CCN(C(c3cnnn3C)=O)CC2C)C)CCCC1 C=C(C)CN=C(NCc1nc2c(s1)CCCC2)NCC1(C)CCCOC1 N1(C(C(C)OCC)=O)CCOC(CC(=O)NCc2csnc2C)C1 C(=O)(C(CCC)CC(C)C)NCCCN(C(=O)CC1CCOC1=O)CCC C1(NC(C(C)Cc2ccnn2C)=O)CCN(C(=O)C(C)(C)C2CC2)CC1(C)C N1(C(CCCCCN(C)C(C2(C)CCCO2)=O)=O)CC2CCC(C1)N2C C1(C(=O)NCc2csc(Cl)c2)(OC)CCN(CC2CCOC2)CC1 c1(C(=O)NCC2CC(NC(C3N(C)C(=O)OC3)=O)C2)cnc2ccoc2c1 C1(N(CCOC)C(C2CS(=O)(=O)C2)=O)CCN(C(=O)C(C)C(C)C)CC1 c1(N2CCCC(CC#N)C2)nc(=NC2CC2)[nH]c2cc[nH]c12 c1(CNC(C2N(c3nc(C)c(F)cn3)CCOC2)=O)ccc2nc[nH]c2c1 C1(C(=O)NC(C)Cc2cc(C)[nH]n2)(COC)C=CCN1C(C1CC1(C)C)=O C=C(Br)CC(=O)N(C)CC1CCCN1C(c1ccnn1CC(C)C)=O Cc1ccc(Br)c(C(=O)NC2CC23CC(NC(c2cc(Cl)c[nH]2)=O)C3)c1 N(C(=NCc1n[nH]c2ccc(Cl)cc12)N1CCN(S(C)(=O)=O)CC1)C(CC)CC c1(NC(CCNC(c2c(CC)onc2C)=O)C)ncnn2c(Br)ccc12 N1(C(CCC(CN(C)C)NC(C(CC#C)(C)CC)=O)=O)CCc2cnccc2C1 c1(C(=O)OC)ccncc1C(=O)NCC1CCN(C(C2CC2(Cl)Cl)=O)CC1 N1(C(c2ccc(CC)cn2)=O)Cc2ccccc2CC1CNC(=O)C(Br)=C(C)C C1(C(N2CC3C(CNC(c4coc(Cl)c4)=O)C3C2)=O)CC2CC1C1C2C1(F)F C(CCC(C)C(=O)NC1CC(C)N(C(c2cccc(CN=[N+]=[N-])c2)=O)C1)OC Cn1nc(C2CC2)nc1CC(=O)NCCC1CN(C(C2COC(=O)O2)=O)CCO1 c1(C(=O)NC2(COC)CN(C(C3C(C4CC4)C3)=O)C2)sc(OC)nc1Cl.CC N1(C(COCCC#C)=O)CCN(C(C2CC(C)OC(C)C2)=O)CC1C(F)F N1(C(C(C)(N(C(c2c(CC)noc2)=O)C)C2CC2)=O)CCCC(C#N)C1 C1(NC(C#CC(=O)O)=O)COC2(CCN(Cc3c(F)ccc(O)c3F)CC2)C1 c1(C(=O)NCC(C2CC2)NC(C(COC)N(C)C)=O)cnn2c1NCCC2 C(=O)(C(CS(C)(=O)=O)c1ccccc1)NCCC(=C)CNC(=O)Cc1cnns1 c1(COC)cccc(C(=O)NC(CNC(c2cnc(C(N)=O)cn2)=O)CO)c1C N1(C(c2n(C)c(Cl)nc2)=O)CC(CNC(C2CC2Cl)=O)C(F)(F)C1 C1(C(=O)N(CC(O)CF)C)(CC)CCCN1C(c1ccncc1Cl)=O C1(NC(CN(c2ccccc2)C)=O)COCCN(C(C2(S(C)(=O)=O)CC2)=O)C1 c1(C(=O)NC)cccc(C(=O)NCC(CNC(C2CCC2(C)C)=O)OC)n1 N1(c2snc(C)n2)CC2CC(NC(c3ccncc3Cl)=O)CC2C1 C1(C2CCN(C(=O)CS(=O)CC)CC2)(NC(C2C(C(C)C)(CC)C2)=O)CC1 C(CN=c1nc2c(cnn2C)c(NC(c2ccc(C)cc2)C)[nH]1)OCCCC N1(C(C2(CNC(COC(C)(C)C)=O)CCC2)=O)CC2CCC1C2 N1(C(C(C)O)=O)CC(NC(c2ccncc2N)=O)C(N2CCCC2=O)C1 Nc1c(C(N2CCCC2CCNC(=O)CC23CCCC2C3)=O)ccnc1Br c1(C(N2C(CNC(CCC(=O)NCC)=O)CCC2)=O)cc2c[nH]nc2cc1C CCC(C)(O)C(=O)N1CCC(CCN2CCN(C(c3cccnc3)=O)CC2)CC1 c1(C(=O)NCCC(=C)CNC(=O)C(CC)=CC)ccc(-c2ccsc2)nc1C c1(CC)ccc(C(N2CCC(CNC(C3CCCN(C(=O)NC)C3)=O)C2)=O)cn1 N1(C(c2c(C)cc(Br)cn2)=O)CCOC2CN(Cc3cccnc3C)CC12 C1(NC(=O)Nc2c(C(=O)OC)c(C)nn2C)CCc2nc(=N)[nH]cc2C1 c1(C(=O)NC2CC(NC(c3nc(C(C)OC)oc3)=O)C2)n[nH]c(C)c1O CC1CN(C(C23CCC(CC2)C3)=O)CCC1NC(=O)CNC(C1CCCCC1)=O C12(c3cn(CC(=O)NCC4(COC)CCCCO4)nn3)CCC(CO)(CC1)CO2 C1(c2ccccc2)(C(C(=O)N(C)C)N(CC(C)O)CC(=O)NC2CC2)CCCC1 C1(CNC(C=CCCC)=O)CN(C(c2cc(C)n(CC)n2)=O)CCC1C c1(C(=O)NCC2C(C)CN(C(=O)CC3(O)CCOC3)C2)cc2n(n1)CCC2 N1(C(c2c(CSC)cccn2)=O)CCC(C)CC1CNC(=O)Cn1ccnn1 N1(C(CCC(=C)Br)=O)CC(NC(=O)CCc2cnn(C)n2)CCC1C c1(C2(CN(C)C)CCC2)cn(CCC(=O)NCC(c2ccccc2)(C)C)nn1 c1(C(=O)NC(C)(CNC(=O)COCCF)C2CCC2)cc([N+](=O)[O-])n[nH]1 CC1(C)CC(CNC(C2CCN(CCO)C(=O)C2)=O)N(C(=O)CC2CC23CC3)C1 N1(C(Cc2nc(C)oc2)=O)CC=C(C(C)(C)C(=O)Nc2ccc3n[nH]cc3c2)C1 C1(NC(c2cc(C)ncn2)=O)CS(=O)(=O)CC1NC(c1cc(C#N)on1)=O C1(CC(=O)N(C2CCN(C(c3c(C)nc(COC)s3)=O)C2)C)CCC(=O)NC1=O C1(C(N(C)Cc2nc(C)[nH]n2)=O)CC(=O)CN1C(=O)CC(=O)OC(C)(C)C C1(NC(=O)CNC(C2CCC=CO2)=O)CC(=O)CN1C(=O)CCCN1CCCC1 C1(NC(C(C)=C2CCCC2)=O)CCN(C(=O)C(=O)NCC2CC2)C1C N#Cc1ccsc1C(=O)NCC1(C(C)(C)O)CN(C(=O)CC2CCC2C2CC2)C1 C1(CNC(COCCCC)=O)CC2(CC2)CN1C(=O)C(c1ccc(F)c(C)c1)=O c1(C(C(=O)N2CC(N3CCN(C(=O)CCF)CC3)C2)(F)F)ccc([N+](=O)[O-])cc1 c12cnn3c1CCCN3C(=O)C2.c1(C2(C(=O)OC)CNC2)ccc(Cl)cc1 C1(CC(N2CCC(F)C2)=O)CCCN(C(c2cc[nH]c2)=O)C1 c1(NC)ccc(C(=O)N(CC(O)CN(C)C(c2oc(C(F)F)cc2C)=O)C)nc1 Cc1[nH]nc(Cl)c1C(=O)NCC(C(C)(C)C)NC(c1c[nH]nc1C(C)C)=O C1(NC(C2OCC(C)C2)=O)CCOC12CCN(C(c1cccc(N(C)C)n1)=O)CC2 C=CCCC(CC(C)C)C(=O)NCC1(C)CCCN1c1ncc2ncnc-2[nH]1 c1(C(=O)NC2CCC(NC(=O)CCc3cnc(O)[nH]3)C2)ccccc1[N+](=O)[O-] N1(C(C(C)OC2CCCC2)=O)CCN(C(c2nncn2C2CC2)=O)CC1 C1(CNC(C2CCCC23CCC3)=O)CCCC2CN(C(=O)CC3CCSC3)CC12 C(=O)(C(C)C(C)C(C)(C)C)N1CC(CCNC(c2cccc(C)c2Cl)=O)C1 Cc1ccc2sc(NC(C3(C)CCCN3Cc3cncn3C)=O)nc2c1 c1(C(=O)NC(CNC(c2ncc[nH]2)=O)CO)cc(C(F)(F)F)ncn1 N1(C(c2cn(-c3ccccc3Br)nn2)C(=O)NCCC#N)CC2OC(=O)OC2C1 c1(CC(=O)NCCC2(O)CN(C(C3CCCS3)=O)C2)cc(F)cc(Br)c1 C#CCC(C(=O)N1CCCC1CN(C(c1ccnc(CCC)c1)=O)CC)C1CC1 CON1CC(C(N2CC3CC2(C(=O)NCc2cccc(O)c2F)C3)=O)CC1=O C(COc1ccccc1)(C(=O)N1CCC(CCNC(c2nocc2Cl)=O)C1)OC c1(C(N(C(CNC(c2cc(OC)nn2C)=O)C2CC2)C)=O)cnn2cccnc12 N1(C(CNC(=O)COCC=C)=O)CCC(CC(=O)NC(C)CNC2CC2)C1 Cc1[nH]c(C)c(C(=O)NC(c2ccc(F)cc2)CNC(=O)CCCN(C)C)c1C S(=O)(=O)(c1ccc(N2CC3CCC2CO3)cc1Br)N1C(CC)COC(C)(C)C1 C1(C(N2CC=C(C)C2)=O)CC(NC(C2(C(C)(F)F)CC2)=O)CCO1 c1(C(=O)NCC2(CCNC(C(COC)COC)=O)CC2)nc2sc(C)cn2c1C C(N=c1[nH]nc(-c2ccsc2)s1)C1C(=O)OCC1 C1(NC(C2CCN2C2CCCC2)=O)CCCCC12CCCN(C(=O)CCC(F)F)C2 O=C(C#Cc1ccccc1)N1CC2CCC(C1)N2Cc1c(I)ccnc1Cl CCCC(C(=O)NC(C(=O)NCCOCC(=O)OC)C1CCC1)C(C)C S(=O)(=O)(c1cc(C(F)(F)F)ccc1NC1COCC1F)N(C(CC)CO)C c1(C(=O)NC23CN(C(C4C(C)C4C)=O)C(C2)C3)ccc2ccccc2n1 C1(C(=O)NCC2CC(F)(CNC(CS(C)(=O)=O)=O)C2)OCC2COCCC12 Cc1cc(F)cc(C(=O)NCC(C)CN(C)C(c2ccc(CO)c(Cl)c2)=O)c1C c1(-c2nc(C(N3CCC(c4ccc(F)nc4)C3)C)on2)ccnc(Cl)c1 C1(OCC)CC2(C1)CC2C(=O)NC1(C)CCN(c2cc(C(=O)OC)ncn2)C1 c1(C(=O)NCC2(F)CN(C(CC3CCCN(C)C3)=O)C2)n[nH]c2c1CCSC2 C(=O)(CCC(=O)NC(C1(O)CN(C(=O)CCc2cc[nH]n2)C1)C)NCCC c1(C(=O)NC2CCN(CC(c3ccccc3)OC)CC2C)nc2cnccc2s1 C1(OC)CCn2cc(CNC(C3(C(F)(F)F)CCN(C)C3)=O)nc2C1 C=CC1(CC(N2CC(CNC(c3ccc(SC)o3)=O)(COC)C2)=O)CCCCC1 Cc1nc(F)ccc1C(=O)Nc1nccnc1C(N)=O.C12(CC1)C(=O)NC2 N1(CC)CC(C(=O)NC2CC(C)(NC(=O)CC(c3ccc(Cl)cc3)O)C2)CC1=O CCCCCC(=O)NC1CC(CNC(=O)Cc2ccc(C)nc2)C1(C)C N1(C(c2c(C)cco2)=O)CCC2C(CCCN2C(=O)Cn2cccc(N)c2=O)C1 C1(NC(c2cccc(N3CC(C)(C)C3=O)c2)=O)CN(C(=O)C(F)(F)F)C(C)(C)C1 c1(C(=O)NC(C(C)NC(c2nc(CC)oc2C)=O)C)c(Cl)ccnc1C N1(C(C2CC(C)N(C)C2)=O)CC2CC(NC(=O)C(CO)C(F)(F)F)CC(C2)C1 CN1CCOC(C(=O)NC2CCCC2CN(C)C(C2(CO)CCC2)=O)C1 c1(C(=O)NCC2C(C(=O)NC(C=C)CO)OCC2)cc(O)ccc1F C1(NC(C2(COC)CCCO2)=O)CN(C(=O)Cc2ccc(O)cc2)C2CC12 N1(C(Cc2scc(C)c2)=O)C2CCC(C2)C1CC(=O)NC1CC1(C)C(F)F C(c1ccc2c(c1)CCO2)=CC(=O)N(CCOC)CCNC(=O)C(C)CO c1(C(=O)NC2CC(NC(c3cn(C(F)F)cn3)=O)C2)ccc(Cl)o1 c1(C(N2C(C(C)NC(C3CCC(C)(C)O3)=O)CCC2)=O)ccc2nc(O)[nH]c2n1 C1(C2CC2)(C(N2CCC(O)(CCNC(c3ccoc3Cl)=O)C2)=O)CC=CC1 Cn1cc(-c2ccccc2CN2Cc3cccc(F)c3C2)c2ccccc12 N1(C(C(C)NC(N)=O)=O)CCC(NCCCC2CCCCC2)C(C)C1 c1(C(=O)NCC2(F)CC(CNC(C(=Cc3cccs3)C)=O)C2)cnc(C)n1C c1(C(N(C2CCN(C(=O)C(=Cc3cccs3)C)C2)CC)=O)cc(C)sn1 C(c1ccc2ccccc2c1)=CC(=O)NCC1CCCN1C(=O)C=CC1CCC1 C1(NC(=O)CC2CCCCCC2)CN(C(c2ccc(F)c(F)c2)=O)CC1C1CC1 NS(=O)(=O)C1(C(=O)NCCN(C(C2CCCNC2=O)=O)C2CC2)CCC1 c1(C(C(=O)NCC(CC)NC(c2cncnc2)=O)N(C)C)ccccc1 N1(Cc2nc(N(C(C)=O)C(C)C)sc2)CCC(C2CC2)(C(=O)O)C1 c1(C(=O)NCCCCCCNC(C2C(C)(C)C2(C)C)=O)ccn2c1CSCC2 c1(CC(=O)NC2CC(C)(NC(C(C(C)C)c3ccccc3)=O)C2)ccccc1C#N CCC(CC)(CN=c1nc(N(CC(=O)NC)C)c2c([nH]1)COC2)C(F)(F)F c1(N(C)Cc2n[nH]c(=N)s2)cc(S(=O)(=O)NC2CCCSC2)ccc1C#N C1(N(C(C(CC)OC2CCCC2)=O)CC)CCN(C(c2cnns2)=O)CC1 C1(NC(CCCOCC=C)=O)CCCN(C(=O)C(C)(C)c2ccnn2C)CC1F C1(CC(=O)NCC2CCCN2C(=O)CC2CC=CC2)CCC(=O)N1 N1(C(C(C)SCC)=O)CCC(NC(=O)C(C)CC(C)CC)C12CCCC2 O=C(CC1=Cc2ccccc2S1(=O)=O)NC1CCC1CNC(=O)CC1CCCO1 N1(C(c2nccc(C)n2)=O)CC2(C1)SCCC2NC(=O)C(n1ccc(C)n1)C C#Cc1cc(C(N2CCN(C(c3csc(Cl)c3)=O)C(C)C2)=O)cc(N)c1 CC(CCOC(C)(C)C)N=c1nc2c(ncn2C)c(NCCCSC(F)F)[nH]1 c1(C(=O)NC(C)(CNC(C2CCCCC(=O)N2)=O)CO)cncc([N+](=O)[O-])c1 N1(C(CC2(COC)CC2)=O)CCC(C)(NC(=O)Cn2ccnc2C)C1 CC1CCCN(C(C2CC(N(C)C)C2)=O)C1CNC(C12CCC(CC1=O)C2)=O N1(C(C(N2CCC(C)CC2)=O)=O)CCCC(C)(C)C1CNC(C1CC1C(C)O)=O C1(OCC(C)C)CC(NC(c2cncc(C(C)(C)C)c2)=O)C1(C)C c1(CN(C(=O)CCCN2CCCC(CC(=O)O)C2)C(CC)C)ccc(CO)cc1 C1(c2cccc(OC)c2Cl)NC(=O)N(C2CC2)C2=C1C(=O)NC(C)C2 Cc1cc(C(=O)NC(CNC(c2cnc(-c3ccsc3)s2)=O)CO)c(C)cn1 N1(C(COCCC(C)C)=O)CCOCC1CNC(=O)Cc1csc(C(C)C)n1 c1(C(=O)NC2CN(C(C3CCC(=O)N3)=O)CC2(F)F)cc(F)c(Br)cc1[N+](=O)[O-] N1(C(c2ccc(CO)cc2)=O)CC2C3CCC(C2C1)N(C(c1csnc1Cl)=O)C3 N1(C(C2C(NC(C3(CC)CCCO3)=O)CCCCC2)=O)CCC(O)CC(C)(C)C1 N1(C(c2c(C#C)c[nH]n2)=O)CCC2CN(C(c3sc4nccn4c3C)=O)CC2C1 C(CC(CC)C(=O)NCC(C)NC(c1nccc(OC)c1F)=O)=CC C(=O)(C(O)C(C)(C)CC)NCCC1CN(C(C2(CC#C)CC2)=O)CC1C N1(C(c2ccc(OC(F)(F)F)cc2)C(=O)NCCCCCC)CC(O)C(C)(C)C1 C1(CC#C)(C(=O)NCCCNC(C2CC2C(F)F)=O)CN(C(=O)OCC)C1 C12(C(=O)NC(C(=O)NCC)C)CC(CO)(CN1C(=O)Cc1ccsc1C)C2 N12CCC(C)(C)C1C2.c1(C(=O)OCC)ccn(C2CCC2)n1 CCCS(=O)(=O)CC(=O)N1CCC(N(C)C(c2cnc(C(C)C)s2)=O)C1 N1(n2c(C(=O)OCC3N(C)C(=O)CC3)ccc2)Cc2ccccc2C1 C(=O)(N=c1ccn(C2CC2)[nH]1)C12C(NC(c3ccc(Cl)cc3)CC)CC(CC1)C2 C1(C(N2CC(CCNC(CCC)=O)C2)=O)CN2CCN1CC2C CCC(C)(C)C(C)NC(=O)CC(C)NC(=O)Cc1ccnn1C c1(C(N2CCC(CCNC(CC3CN(C)C3)=O)CC2)=O)cc2c(F)cccc2[nH]1 N1(C(C(C)NC(C)=O)=O)CC(N(C(=O)Cn2nc(O)ccc2=O)C)C2(CC2)C1 CC1CC2CC2CC1C(N1CC(CNC(=O)CN2CCOC2=O)C1)=O C(CC(C(=O)NC(C1CCCC1)C)NC(=O)C(=CC1CCCC1)C)OC c1(C(=O)NCC2CCN(Cc3cnc(Br)s3)C2)ccc2c(c1)CCNC2 C1(CC)C(NC(c2ccc(OC)s2)=O)CCCN1C(=O)CCC1CCOC1 c1(C(=O)Nc2c(OC)cccc2OC(F)F)cnc2c(Br)cccn12 Cc1ccc(OCC(=O)NCC2CN(C(C34COC(C(C)C)(C3)C4)=O)C2)cc1 C1(C(=O)NCC2CC(NC(c3cnc(-c4cccs4)s3)=O)C2)CCCC1O c1(C2(OC)CC2)ccc(CNC(=O)CC(O)C2CCCC2)cc1.C12(CC1)C(=O)N2 CC1(C)CCN(C(c2cc(C(F)F)cs2)=O)CC1CNC(C12CCN(CC1)C2)=O N1(C(C(C)=CC)=O)CC2(CNC(C3CCC(=O)N3C(C)C)=O)CCC1C2 Cc1nc(NC2CCN(C(C3CCOC(C)C3)=O)C2)cc(Cl)n1 N1(C(CC(C)OC)=O)CCC2(CCCC2CNC(c2n[nH]c(C3CC3)n2)=O)CC1 CC1CN(C(=O)CC#N)CCN1C(c1cnc(N(C2CCCCC2)C2CCC2)s1)=O CC1(CC(=O)NC2CC2CNC(=O)C(c2ccc(Cl)nc2)(C)C)CCS(=O)(=O)N1 CCCCCCC(F)C(=O)N(CC(C)NC(c1ccc(CCC)s1)=O)CC CC(C)CC(O)C(=O)N1CCC(C(=O)NCCC2CCCC2(C)C)C(C)C1 c1(C(N2CC(O)(CNC(CC(CN(C)C)(C)C)=O)C2)=O)c[nH]c2cc(Cl)ccc12 N1(C(C(C#N)=CC(C)C)=O)CCC(C)C(NC(C2CCC(N=[N+]=[N-])C2)=O)C1 C1(n2c(SC)ncc2)CN(c2ccc(S(=O)(=O)NC3CC3)cn2)CC12CCOCC2 C=CCC(C(=O)NOCCCOC)NC(=O)CCCN(C)C c1(CNC(C2COCCN(CCC(=O)OC)C2)=O)noc2ccccc12 Cc1ccc(F)c(C(N2CC3(CCN(C(C4(C)CCOC4C)=O)C3)C2)=O)c1N c1(C(=O)NC2C(C)CCN(C(c3ncccn3)=O)C2)cccc2c1CCC2 C1(CNC(C(C(C)C)SC)=O)CC(C(C)(C)C)CCN1C(c1cscc1F)=O N1(C(COC)=O)CC2CC(NC(=O)CCOc3ccc(F)cc3)CC2C1 c1(CC(N2CC(CC=C)(NC(C3(F)CCOC3C)=O)C2)=O)ccc2c(c1)OCO2 C1(CNC(c2n(C(C)C)ncc2)=O)CCC(C)N(C(c2cc(CCO)on2)=O)C1 C(=O)(C1=C(C)OCCC1)NC(CC)CNC(c1cncc(C(C)(C)C)c1)=O c1(C(=O)NC(C(C)C)CNC(=O)C(F)(F)C(C)O)cc2c(Br)cccc2[nH]1 Cc1nc(C(=O)N(C2CCC(NC(c3ccc(NC=O)cc3)=O)C2)C)c(C)o1 Cc1nccc(C(=O)NC2CC(F)(F)CC2NC(=O)C(C(C)C)N(C)C)c1C C1(CNC(C2CC(=O)NC2)=O)(NC(C2C=CCC2)=O)CC2CCC1CC2 c1(CC)noc(CC)c1CC(=O)NCCC1CCCN(C(c2nonc2N)=O)C1 C(C(=O)NOCc1nc[nH]n1)C1CN(C(C=CCN(C)CC)=O)C1 CCC(CC(=O)NCC1(NC(=O)CCCC(OCC)OC)CCC1)C(C)(C)C N1(C(C2(CC)COC2)=O)CC2COCC2(C(=O)NCCCCC(C)(C)C)C1 CC1CN(C(=O)CNC(c2ccncc2)=O)CCC1NC(=O)C1=C(Cl)CCC1 N1(C(CCN(CC)CC)=O)CCCC(CCNC(c2ccncc2C(F)F)=O)C1 C1(CNC(c2c(C#C)c[nH]n2)=O)(OC)CCN(C(=O)C(C(C)OC)N(C)C)CC1 N1(C(c2ccc(CC)cc2Cl)=O)CC2CC(C1)CN(C(=O)C(C(C)CC)OC)C2 C1(C(=O)NCc2c(CC)nns2)CC(CC)CCN1C(=O)Cn1nnc(C)n1 c1(C(=O)NC(C)CN(C(=O)C(F)n2ccnc2)C)c(O)cc(=O)n2c1CCCC2 Cc1cc(C(N2CCC3(NC(=O)Cc4csnc4C)CC3C2)=O)c(Cl)cc1F C12(C(=O)NCCC3(C)CCN(C(=O)CN4CCNC(=O)C4)C3)CCCC1C2(F)F N1(C(c2c(CC)cc[nH]2)=O)CCCC(CNC(=O)COC2CCOCC2)CC1 C(C(C)(O)CCO)NC(C(C1(O)CCCCC1)NC(C(C)CC1CCC1)=O)=O c1(C(=O)NCC2(NC(c3cocc3C=O)=O)CC2)ccc(SC)s1.CCSC C=C1CC2CCCC(C1)N2C(=O)CCC(C)NC(=O)C(C1CCOCC1)C C1(CC(=O)N(C)Cc2ncc[nH]2)CCCN(C(C2CC(O)CN2C)=O)CC1 Cc1ccc(CCCC(=O)NCC#CCNC(=O)CC(C)C)cc1 Cc1cncc(CNC2CCC(CNC(c3n[nH]c(C)n3)=O)CC2)c1 C(=O)(C(O)C1=CCCCC1)N(C(CNC(C1CCCN1C(N)=O)=O)C1CC1)C C1(NC(c2c(CC)[nH]cc2)=O)CCC2CC1CN2C(C1CCSC(C)C1)=O N1(C(CCC#C)=O)CCC2CCN(C(=O)CCC(=O)NN(C)C)C2C1 CC1CCCCC1C(=O)N(CCCC(=O)N1CC(C#N)C1)C c1(NC(=O)NCCCC(=O)OC(C)C(=O)N2CCCC2)nnc(O)nc1O c1(-c2cnc(CC(=O)NCc3ccnc4[nH]ccc34)nc2)c[nH]c2cnccc12 c1(C(N(C(CNC(C=C(COC)C)=O)C2CC2)C)=O)nc(C)c(C)nc1O C1(CNC(CC(C)NC(N)=O)=O)CCN(C(=O)C(=O)NCC2CC2)C12CC2 CCC(C(=O)NC1(COC)CCN(C(=O)CSSC)CC1)C(C)O C1(NC(CC2C(C)CCO2)=O)CCC2CCN(C(=O)CCC3CC3(Cl)Cl)C1C2 C1(C(N2CCC(COC)(NC(=O)CC3CCOC3)C2)=O)CCC2(CCC2)O1 c1(SC)ccc(C(=O)OC(C)Cc2cccc(C)n2)cc1Br C1(C(=O)NCC(CO)NC(c2ncc(C)nc2)=O)Cc2ccccc2C(=O)O1 N1(SCCOC(N2CC(F)(F)C2)=O)CC=CC1(C(F)(F)F)CNC(=O)OC(C)(C)C C(C1COc2ccccc21)c1nn(C(C2CCCO2)C)c(-c2nocc2Cl)n1 C1(C(N2C(CCN(C)C)CCC2)=O)(CNC(c2cnc(O)o2)=O)CC2(CC2)C1 C(c1ccccc1F)=CC(N1C(CCNC(C(C)OCC(C)C)=O)COCC1)=O C=CCC(CC)C(=O)NCc1nocc1C(=O)Nc1c(C)noc1C CC(C)(O)C(C(=O)NCCCCC(F)(F)F)NC(=O)Cn1cccn1 c1(C(N2CCN(C(C(CCC)N(C)C)=O)C(CC)C2)=O)c[nH]c2ccc(O)cc12 C1(CNC(C2CC(OC)C2)=O)CC(F)CN1C(=O)C(C)c1cscn1 c1(OC)ccc(F)c(CC(=O)NC2CC2CNC(C23COCC2C3)=O)c1 S(=O)(=O)(c1cccc(C(N2CCCC(CNC(=O)C(C)N(C)C)CC2)=O)c1)NC Cc1ccnc(C(=O)NC2CCCC(CNC(c3c(C)ncnc3C)=O)C2)c1N CC(C)CCCC(C)C(=O)N1C2CCC(C(=O)NCC34CC(CCO3)C4)C1CC2 Cc1c(C(=O)NC(C)(C(=O)NC2CN(C(=O)C3CC3)C2)C2CC2)cccc1C#N N1(C(CCC(C)OCC)=O)CC2(CCN2C(=O)Cc2ccoc2)C1 c1(CN2CC3C(C(N4CCCOCC4)=O)(C3)C2)ccc([N+](=O)[O-])cc1 C1(CNC(c2cc(CC)ncn2)=O)CCC(C)CN1C(c1cc(C)on1)=O C1(C(=O)NCCOCCNC(C2(CO)COC2)=O)CC(n2cnnc2)C1 N1(C(c2n(C)ncn2)C(=O)NCC2CCOC2)CC2CS(=O)(=O)CC2C1 N1(CC(=O)NCCN(C)C(c2ccnc(C(C)(C)C)c2)=O)C(=O)CNC1=O C1(NC(c2cc(CC)nn2C)=O)CCC2CC1CN2C(c1ccnc(Cl)c1F)=O c1(C(N2CCC(CN(C(C(C(=O)OC)(C)C)=O)C)C2)=O)ccc2c(n1)CCCC2 c1(C(=O)NCc2cc(C(=O)NC(CC)(C)C3CC3)n(C)n2)ccc(C#N)cc1 C1(N(C(=O)C(c2ccc(F)cc2)(F)F)Cc2cn(C)nc2)CCNCC12CC2 C(=O)(C(O)C(F)(F)F)NCC1C2CN(C(c3c(C)[nH][nH]c3=N)=O)CC21 N1(C(c2n(C)ncc2)=O)CC2(C)CC1(C(=O)NCC1(Cl)CCC1)C2 CCC(C)C(C(=O)N1CCCC1(C)CCCO)N(C(=O)Cc1ccc(C)s1)C N1(C(C2CN(C(C)C)C2)=O)CC(CNC(c2cnco2)=O)CC(C)(C)C1 C1(C(=O)NC(CCN(C(COC(CC)CC)=O)C)C)CCc2nn[nH]c2C1 c1(C(N2CC(CC(C)NC(=O)Cc3c[nH]nc3O)C2)=O)ncoc1C(C)(C)C Cc1cc(C(N2CC(CC(C)NC(C3CCCSC3)=O)C2)=O)c(Cl)cc1N C1(N(C(CCN(CCC)C)=O)C)CCN(C(=O)CCc2cc(C)no2)C1 Cc1cnc(C(=O)NCC2CC(O)CN2C(C2CCN(CC(C)C)CC2)=O)nc1 C1(NC(C(C)OC)=O)CCC2(CC1)CC(NC(c1ccc(F)c(F)c1F)=O)C2 CC1CN(C(=O)CC2N(C(=O)C=C3CCOCC3)CCC2(C)C)C(C)C1C Cc1ccc2c(N(C)Cc3ccnn3C)nc(=NC3CSCCSC3)[nH]c2c1 N1(C(CC2(OC)CCC2)=O)CC2(CCC(NC(=O)C(C)COC)CC2)C1 c1(OC)ccnc(C(N2CCC(OCCNC(C3(Cl)CC3(F)F)=O)C2)=O)c1 c1(C(N2CCN(C(=O)CC3(C(F)(F)F)CC3)C(CF)C2)=O)cccc2[nH]ccc12 C#CCCCC(=O)N1CCCCC1CCCNC(=O)C=CC(C)(C)C N1(C(CC2CCCC(C)O2)=O)CC=C(CNC(C2CCC3CCC2O3)=O)CC1 Cn1ncc(C(F)F)c1C(N1CCOC(CNC(=O)C=CC2CCOCC2)C1)=O N1(C(CCC2C(C)(C)C2)=O)CCN(C(=O)Cc2cccc(Cl)c2)CC1CCO C(=O)(C(=O)N=S(C)(C)=O)NCCN(C(C=Cc1n(CC)ncc1)=O)CC1CC1 C1(CC)CN(C(c2c(OC(F)F)cccc2F)=O)CCN1C(C1COC(=O)C1)=O Cc1cccc2c1OC(C(=O)N(C)CC1(NC(=O)Cn3nccn3)CC1)C2 N1(C(C(CC)C#N)=O)CC(NC(c2ccccc2C(C)O)=O)C2CCCCC12 C(=O)(C(F)C(F)(F)F)N(C(C)(C(=O)NC1(C)CC1)C1CC1)C N1(C(CCCN(C)C)=O)CCC2CN(C(=O)Cc3cn[nH]c3)CCC2C1 C1(O)(CN2C(CNC(=O)COCC3CCCO3)CCC2)CCc2ccccc2C1 C1(C(=O)NC2(CNC(c3ccsc3Br)=O)CC2)CC12CC2(F)F N1(C(C(CC)Cc2ccccc2)=O)CCN(C(c2csc(C)c2)=O)C(C2CC2)C1 CC(C)(CNC(=O)CC1CCC(=O)N1)CNC(C1(n2cccc2)CCCC1)=O C1(CN(C(=O)CCC2CCCCO2)C)CCN(C(=O)CSCC2CCCO2)CC1 C1(NC(c2ccc(CC)cn2)=O)C(C)CN(C(=O)C(F)=C2CCCC2)CC1C c1(OC)cc(F)c(-c2ccc(C(C)NC(c3cccc(I)c3F)=O)cc2)cc1F N1(C(c2cc(CC)no2)=O)CC=C(CC(=O)NCCCc2nncs2)CC1 C1(CC)CCCC(OC)N1CC(c1ccc(-c2ccccn2)nc1)=O CCS(=O)(=O)C1CN(C(=O)NC2CCN(c3cccc(OC(F)(F)F)c3)C2)C1 C(=O)(C(CC(F)(F)F)c1ccccc1)N1CC(O)(CNC(c2ccc(F)o2)=O)C1 c1(C(=O)NC23CC(C(=O)NCCCCCCCCO)(C2)C3)ccn2ccccc12 c1(CN2CCC(C#N)(NC(C(C)NC=O)=O)C2)ccc2nc(O)[nH]c2c1 N(C=CC(=O)C(F)(F)F)C(C1CCCN(Cc2ccc(Br)c(Cl)n2)CC1)=O C1(NC(CC2CCN(CCC)C2)=O)CN(C(C2(C)CNC(=O)C2)=O)CC1C(F)F N1(C(C2ON=C(CC)C2)=O)CCC(C)(NC(=O)Cn2ncc(Cl)c2C)CC1 C(=O)(C(C(C)(C)O)NC(=O)CCC1CCOCC1)N1CCCC(OC)C1 c1(-c2c(C(=O)NC)cccc2)cccc2[nH]c(C(=O)Nc3cc(O)ncn3)cc12 Cc1cn2cc(C(N3CCC3CNC(c3ccc(Cl)cc3C(F)F)=O)=O)nc2s1 O=C(C=C(Cl)Cl)NC1CCC1NC(=O)CNC(c1cccnc1)=O N1(C(C=C(CC)CC)=O)CC2(CCOCC2)C1c1cn(CC2CCC(=O)O2)nn1 C(=O)(C(O)CC(N)=O)NC(CC)CN(C)C(c1cnn(C)c1C(C)C)=O c1(C(=O)NC(C(=O)OC)CCF)ccc2c(c1)OCC(=O)N2 C1(CNC(C2(CC=C)CCCN2C(c2oncc2CC)=O)=O)C2CCCCCC12 C1(NC(C(C)=C(C)C)=O)CCC(N(C(=O)C(O)CN(C)C)C)CC1 C1(C(=O)NCCC2CCN(C(c3[nH]c(CC)c(Cl)n3)=O)CC2)CC1C1CCCC1 N1(C(c2ccn(CC)n2)=O)CCN(C(c2ccc(C)cc2OC)=O)C(COC)C1 N1(C(C(CCOCC)NC(=O)C(n2ccc(C)n2)C)=O)CC(F)CC(F)C1 Cc1csc(C(=O)NCC(C)NC(c2c(C)n[nH]c2C)=O)c1Br c1(OC(C(=O)OC)C)cccc(Cc2csc(-c3ccccn3)n2)c1 S(=O)(=O)(c1ccc(Cl)cc1)N(C(C1CN(CC)C(=O)N1)=O)C(C)C N1(C(C(c2ccccc2)=O)=O)CC2CC1C2NC(=O)C=CC1CCOCC1 N1(c2ncnc(C(C3CCOCC3)=O)c2F)CCc2ccc(Cl)cc2CC1 Cc1cc(N)ccc1C(=O)NCCCOCCCNC(=O)C(c1ccnn1C)O c1(C(=O)NC2CCCN(C(CC3CCCC(C)O3)=O)C2)ccc(F)c(F)c1 N1(C(c2c(OC)cncn2)=O)CC(NC(=O)CC=Cc2ccccc2)CC(O)C1 c1(NCC(CNC(c2cncc(C)c2)=O)C)cc(O)nc(=O)n1C c1(C(N2CCC(O)(C(C)NC(c3cccc(=O)o3)=O)C2)=O)cc2cc[nH]c2cn1 c1(N2CCCC(C(C)NC(=O)CCOCC3CC3)C2)ccc(C#N)nc1 CCCCCCC(F)C(=O)NC1(C2CCN(C(C3CC3OCC)=O)CC2)CC1 C(=O)(C1=CC2(CN(C(c3ccnnc3O)=O)C2)OC1)N1CCC(C)(F)C1 C1(C#N)(C(=O)NC2CCCC(N(C(C=C(C)Cl)=O)C)C2)CCOCC1 n1(CCOC)ccc(=NC(=O)c2ccc(CNC(c3ccc(C)cn3)=O)cn2)[nH]1 c1(C(=O)NCC2CCN(C(C(C)C#N)=O)C2)nnn(C)c1C(F)(F)F Cc1sc2ccccc2c1C(N1CCC2(NC(C3CC34CCC4)=O)CCCC12)=O C12(NC(CC(=O)NCC)=O)CCC(CC1NC(=O)CCC(C)C#N)C2 n1(C(C)C)cc(C(=O)NC(C)C(C)NC(c2sccc2OC(F)F)=O)cn1 C(=O)(CC(C)(C)c1ccc(F)cc1)NC1CN(C(C(c2ccc(F)cn2)C)=O)C1 c1(C(=O)NCC2(COC)CN(C(C(C)OCC=C)=O)C2)c(F)ccc(OC)c1F C1(CN(C(C2N(CC)CCC2)=O)CC)CCN(C(=O)Cc2nncn2CC)CC1 C(=O)(C(F)CC1CCCCC1)N(C(C)CN(C(=O)CCN1CCCC1)C)C1CC1 N1(C(C2(C(C)C)CCC2)=O)CC2(C=C(C(=O)NC3CCOCC3C)CO2)C1 C1(CNC(CC)=O)COCCN(C(=O)C(C)C)C1 CC1OCCN(C(C2(N(C)C)CC2)=O)C1CNC(C1CCC(=O)N1C)=O CC1CCCC(C(N2CC(C)(CCC(=O)NCCn3ccc(=O)cc3)C2)=O)CC1 N1(C(C=C(C)C(F)F)=O)CCN(C(c2cc(C)ns2)=O)CC1c1cccc(F)c1 C1(CNC(c2c(C(C)C)ocn2)=O)C2CC2CN1C(c1cnc(C(N)=O)cn1)=O N1(C(C(=O)NCC)=O)CC2CC2(CN(C(c2cnn(CC(=O)OC)c2)=O)CC)C1 c1(C(=O)NC(CN(C(=O)C=Cc2cncn2C)CC)C)nc(Br)cnc1N C(CC(C)C)(C(=O)N1CC(NC(C2CC3C=CC2C3)=O)CCC1C)OC Cc1nc(C(=O)NCC2(NC(=O)C=Cc3ccnn3C)CCC2)nn1C c1(CNc2cnn(C(CC)C)c2C2CC2)ccc(C)n(C)c1=O C(=O)(C(CC)NC(=O)NC(C)CNc1ccc(CC(C)C)s1)OCC CC1CC(CNC(c2cn(C)nc2-c2ccoc2)=O)CCN1C(c1cnns1)=O C1(CC(C)NC(CN(CCOC)C)=O)CCN(C(=O)C(C)C2CC2)CC1 Cn1cncc1C(N1CC(NC(C2CCCC2n2cccc2)=O)C1)=O Cc1cc(F)ncc1CNCc1cccc(NCC(C)C)c1 Cc1[nH]nc2cc(C(=O)NCC3CCN(C(=O)C=CCF)C3)ccc12 c1(C(C(=O)NC(C)(C)C)N(C(C2(C)CC2)C)C)ccnc(Cl)c1OC CC1=CC2CC(NCC(C)(N)Cn3cccn3)CC(C1)C2 c1(CCC(=O)N(CC(CNC(C2C(C=C)C2)=O)O)C)cncnc1 C(=O)(C(C(C)C)NS(N)(=O)=O)NCC(CCC)NC(c1csnc1C)=O Cc1ccsc1C=CC(=O)NC(C)(CNC(C1CC(=O)N(O)C1)=O)C1CCC1 C12(CCC1)C(=O)NCCN(CCOCC)C2=O.C1(C)(SC)CC1 C(c1cncnc1O)=CC(=O)NCC1CCCN1C(c1n[nH]cc1Br)=O C1(c2cnc(NC)s2)NC(=S)N(c2ccc(Br)cn2)C(C2CCC2)=C1C(=O)OC Cc1ccc(C)c(CC(=O)NCC2CCC2NC(=O)CCNC2CCCCC2)c1 c1(CC(=O)OC)cccc(CN(CC(=O)O)C)c1.c12cn(nn1)C2.N1(C)CCCC1 c1(C(N2CCC(NC(CC3ON=C(C)C3)=O)CC2)=O)nccc(F)c1Cl c1(C(N2CC(CC(=O)Nc3c(SC)cccc3)OCC2)=O)[nH]nc2ccncc12 c1(C(=O)NC(CCN(C(c2c(C)cccc2Cl)=O)C)C)cccc2nc(O)oc12 c1(C(=O)NCC(CC)NC(C2CCCN2C=O)=O)cccnc1N(C)C C#CCC(C(=O)NC1(CNC(c2ccc(CS(C)(=O)=O)o2)=O)CCC1)C1CC1 C=C=C(C)CC(=O)NCCC(C)CCNC(c1ccn(C2CCCCC2)n1)=O c1(CC(C)(C)OC(C)=O)cn(CCCNC(=O)C(F)(F)C2(O)CCC2)nn1 C(C)(C)(C(=O)N(CC1(O)CN(C(=O)CCc2cccn2C)C1)CC)N(CC)CC CS(=O)(=O)CCN=c1[nH]c(=NCC2CN(CC(F)(F)F)C2)[nH]c2cccnc12 CC1(CCNC(C2CC(O)C2)=O)CCN(C(=O)COCc2ccncc2)CC1 CC(N=c1cc[nH]cc1S(=O)(=O)N1CCOC(CF)C1)C1CC1.CCCO C1(C(=O)NCC(C)(C)OCC(=O)NC(C)CS(C)(=O)=O)CC(C2CC2)=NO1 Cc1nnc(O)c(C(=O)NCCC2(CNC(C3(C)CCCOC3)=O)CC2)c1C c1(NC(C2(c3ccccc3OC(F)(F)F)CC2)=O)ncnc(Cl)c1Cl C1(NC(C(C(C)C)OCC)=O)CC2CCC(C1)N2C(C1CC1C(F)(F)F)=O N1(C(C=CCN(C)C(C2SCCS2)=O)=O)CC2CC=CC1C2 C1(CNC(=O)C2=CCC2)CN(C(c2cccc(F)c2C(F)(F)F)=O)CCC1(F)F CC(=O)CCCC(=O)NCCC(C)NC(=O)CC1CCCC(F)(F)C1 c1(C(=O)NC2C(C(=O)NC(CC(=O)OC)C)CCC2)cccc(C(F)(F)F)c1O C#Cc1cccc(C(=O)NCC2CN(C(c3cc(OC)cs3)=O)CCC2C)c1C C(CN=c1cnc(N)c(C)[nH]1)(c1ccc(C)cc1)N1CCOCC1 c1(C(=O)NC(C=CC(=O)NC(COC)C)C)ccsc1OC1(C)CCC1 n1(CC(CC)O)cc(C(N2CC(O)(CNC(=O)CSC3CC3)C2)=O)nn1 c1(NCC(CO)OC)ccc(S(=O)(=O)NC2CCOCC2OCC(C)C)c(Cl)c1 N1(C(c2n[nH]c(C)c2C)=O)CCN(C(c2ccc(-c3cscn3)cc2)=O)CC1C N1(C(CC(CC)N(C(=O)CC2CCCCN2C)C)=O)Cc2cnn(C)c2C1 c1(OC)ncccc1C(=O)NCC1(Cn2cc(CNC(C)=O)cn2)CC12CCC2 Cc1c(C(=O)N(CCNC(=O)C(C)(O)C2CC2)C2CC2)oc(=O)c2ccccc12 C(C)(CC(C)(C)C)(c1nnnn1C1(C)CC1)NCc1cc(COC)on1 Cc1cccc2c1CC(NC(c1cn(Cc3cccnc3)nn1)=O)C2 C1(NC(c2c(CC)ncs2)=O)CC(CNC(=O)CC2(COC)CCCC2)C(O)C1 c1(NCCC(=O)Nc2ccc(SCC)cc2)c(F)c(C)nc2ncnn12 c1(C(N(CCC(=O)NCC(C)(C)COC)CC#C)=O)sc(C)cc1C Cc1nc(O)[nH]c1C(=O)NCC1COCC1NC(C1CC1c1cncs1)=O C1(C(N(CCCNC(C2(C#N)CCCC2)=O)C)=O)CCCCN1N=O N1(C(C(C)C2CCC2)=O)CC2CN(C(c3ccc(NC4CC4)nc3)=O)CC2(C)C1 S(=O)(=O)(c1cnc(NCC2(C)CCS(=O)(=O)CC2)cc1C)NC(C(CC)(C)C)C C(=O)(CCC(F)(F)F)NCCC(CNC(c1cnn(C)c1C(F)(F)F)=O)O c1(C(N2C(CNC(CC3CCCC(OC)C3)=O)CC2)=O)ccc(=O)n(CCO)c1 Cc1ccc(NCCNC(=O)C=Cc2nc(C)co2)c(Sc2ccc(Cl)cc2)c1 Cc1nc2nc[nH]n2c(=O)c1CCNC(=O)CC(N)C(C)(C)C c1(N2C(CNC(Cn3c(CCC)ncc3)=O)CCC2)nccc(SC)n1 N1(C(C2C(C)(C)C2NC(c2cccnn2)=O)=O)CC2COCC2(CO)C1 N12CCC(C(C)C1)NC(=O)Nc1cc(on1)C2=O.c1(OC)ccncc1C c1(C(N2CCN(C(C3C(C=C)OCC3)=O)CC2C)=O)cnn(C)c1S(N)(=O)=O N1(C(Cc2c(C)cccn2)=O)CCOc2ccncc2C1 CCC(C)(C#N)C(=O)NCC1CC2(CC(NC(=O)CCCCC3CC3)C2)C1 N1(C(c2c(OC)cc(C)nc2)=O)CC2=C(C1)CN(C(=O)COCCF)C2 C12(C(=O)NC(CN(C(C(c3c(C)noc3C)C)=O)C)C)CC(CO)(C1)OC2(C)C c1(OCC=C)ccc(NC(=O)N(C)C(C2CC2)C2CC2)cc1C(F)(F)F CC(CCCNC(c1cc(Cl)ns1)=O)NC(=O)CC(c1ccccc1)N(C)C N1(C(CC(CC)CC)=O)CC=C(CC(=O)NCCCOCC(F)F)CC1 c1(N2CCC(OC(CF)(F)F)CC2)nc(N2CCCC(O)CC2)nc2c1CCC2 C(=O)(CC(C(F)F)NC(C1(C#N)CCOC1)=O)N1CC(CC(C)C)C1 N1(C(c2sc(C)c(O)n2)=O)CCC(C)C(NC(C2CCCC(=O)N2C)=O)C1C C1(CNC(C(C(C)C)O)=O)CC2CCC1N(C(c1c[nH]c3cccnc13)=O)C2 CCS(=O)(=O)CCNC(=O)NC(C1CN(C(=O)OC(C)(C)C)C1)C CCCC(CC)CC(=O)NC1CCCN(C(=O)C(C(C)C)NS(C)(=O)=O)CC1 Cc1cc(C(=O)NCC=CCNC(C2CCCCS2)=O)nn1CCO C1(C(=O)N(CCCC(=O)N2CCC(N3CC=CC3)C2)C)(OC)CCOC1 N1(C(C2(C)CC2(F)Cl)=O)CCN(C(c2ccc(O)c(N)n2)=O)CC12CCC2 C(=O)(CS(=O)(=O)CC(C)C)N(C1CCC(NC(c2c(Cl)ccc(C)c2N)=O)C1)C C1(N(C(=O)C=Cc2nccs2)C)CC(O)CN(C(=O)C(C)(C)c2ccsc2)C1 C12(CNC(c3cccc(=O)o3)=O)CC(CN1C(=O)C(c1ccccc1Cl)(F)F)C2 Cc1cc(-c2ccc(NC(=O)CC(C)N(C)C(C)C)cc2)cc([N+](=O)[O-])c1O n1(CC)cc(C(=O)C(=O)N(C2CN(C(=O)C(C)N(C)C(C)=O)C2)C)cn1 C=C(CNC(=O)C(C)SC(F)(F)F)CCNC(C1CCCN1Cc1ccccc1)=O Cc1ccccc1C(=O)NCCn1cc(-c2ccc(C3CC3)s2)nn1 C1(C(=O)NC2(CNC(c3ccc(Br)cn3)=O)CCCC2)CCn2cnnc2C1 N1(C(CC(CC)C2CCC2)=O)CC(CNC(=O)C(C)=C2CCC2)CC12CCC2 N1(CCNC(CCCSC)=O)CCN(C(=O)CCNC2CC2C)CC12CCC2 NC(=O)CCCCC(=O)N1CCCN(C(=O)CNC(c2cccc(=S)n2O)=O)CC1 c1(-c2sccc2)nc(NC2CCC(N3CCOCC3)CC2)c2ccccc2n1 c1(CC(=O)N(CCCOCCN(C(CCC)=O)C)C)c(F)cc(F)cc1F Cc1c(CNC(N2CC(C)CCC2c2cccs2)=O)ccc2nccn12 N1(C(C(C)NC(N)=O)=O)CC(F)(F)CC1CCNC(=O)C=C1CCC(C)C1 c1(C(N2CCN(C3CCC(OC)C3)CC2)=O)cc2c(OC)cc(OC)cc2[nH]1 c12cc(OC)c(OC)cc1NC2=O.C#Cc1cnn(C)c1-c1nc(C2CC2F)no1 CC1COC2(C1)CN(C(=O)C(CO)NC(c1ccn3cncc3c1)=O)C2 Cc1cc(Cl)c(Cl)cc1C(=O)NCC12CC1CN(C(C1CC1C)=O)C2 C(=O)(C#CC1CCOCC1)NC1CCC(N(c2snc(Cl)c2C#N)C)CC1 N1(C(C2N(C(C(C)C(F)(F)F)=O)CCC2(C)C)=O)Cc2cnn(C)c2C1 CCCCC(CN=c1[nH]cnc(Cl)c1C(=O)OC)NC(=O)C(C)(C)CO Cn1nnc2cc(C(=O)NC3(CNC(C4(F)CCOC4)=O)CCCCC3)cnc12 c1(SCC(=O)NCC2(CNC(c3cc(C)ns3)=O)CCC2)ccccc1Br C(C)(C)(CCC(=O)NC(c1cc[nH]n1)C)NC(C(C)SC(C)C)=O c1(C(=O)NC(CC)C(C)NC(C2(CSC3CC3)CC2)=O)oc(CC(C)C)nc1C CCC(CC(=O)N1CCCC1(C)C(=O)NCC1(CC2CCC2)CC1)C(F)F c1(C(=O)NC2C(C)CN(C(=O)C(F)n3cccn3)C2)cc(F)ccc1C(F)(F)F c1(N2C(C)(C)C(NC(C3CC4C(C3)C4(C)C)=O)CC2)nc2cc(F)ccc2o1 CC1CCCCC1(CNC(C1(C(F)F)CC1(F)F)=O)NC(c1cc(CN)cs1)=O c1(C(=O)NC)ccc(OC)c(-c2ccc(CNC(c3ccc(Br)nc3)=O)cn2)c1 O=C(CC(CNC(c1cc(C(F)F)[nH]n1)=O)C1CCC1)NC1(CO)CC=CC1 CCC(CCO)CN=c1[nH]c(=NC(C)c2nnc(CN(C)C)s2)[nH]c2c1CCCC2 C(C)(CCCCNC(=O)C=CC(N)=O)NC(CCSCC(C)C)=O c1(C(=O)NCC(C2CCCN(C(=O)CSC(F)(F)F)C2)(C)O)ncc(F)cc1F c1(OCC(=O)NC2(C3N(C(CC(CC)C)=O)CCCC3)CC2)cccc(C#N)c1 CC(=Cn1ccnn1)C(=O)N1CC(OCCNC(=O)C(C)(C)CC(C)(C)C)C1 C(CC(=O)NC1(OCCCNC(=O)Cc2ccon2)CC1)NC(=O)NC C1(N(C(C(C)OCCCCCC)=O)C2CCCC2)Cc2ccccc2N1 N1(C(C(C(=O)OC)C)=O)CC2CN(Cc3cc(C)nn3C)C2C1 C1(CN2CCCC(CC)(CC)C2)COCC2(CCNCC2)O1 c1(CN2CCC(O)(COC)C2)c(F)cccc1Br N1(C(C)=O)CCC(CC(=O)NCC23CC2CN(C(=O)CC2COCC2O)C3)CC1 C(N=c1cc[nH]cc1S(=O)(=O)NCC1(C)CCCCC1(F)F)C1(OC(C)C)CC1 c1(C(=O)NCCCNC(C2(C)CC2F)=O)cnc2cnc(Cl)cc2c1 C(=O)(C1=CCCCCC1)N1CC2(CN(C(C(C)(O)C)=O)C2)C1.c12nc(no1)C2.N N1(C(c2nccc(C)n2)=O)CCN(C(C2CC2F)=O)CC1CCO c1(NCc2c(Br)cn(C)n2)cc(=NCc2cc[nH]n2)[nH]c(C(F)(F)F)n1 C12(CNC(CC(CCC)O)=O)CN(C(=O)C(C)(C)C(N)=O)CC1CCO2 c1(CNC(C2CCC(NC(CCCC)=O)CO2)=O)ccc(S(N)(=O)=O)cc1 N1(C(C=CCOC)=O)CC2(COC(CNC(=O)CCC(C)CN(C)C)C2)C1 Cc1c(C(N2CC3(NC(=O)C(C)C(F)F)CCC2C3)=O)cncc1N C1(O)(CC(=O)NCC(CN(C(c2c(CC)nn[nH]2)=O)C)C)CCCCC1 N1(C(CC2COCC(C)O2)=O)CCCN(C(=O)Cn2nnc(=N)[nH]2)CC1 c1(C(=O)NC2CC2CNC(C2(Cl)CC23CCC3)=O)cc2c(Cl)cc(Cl)cc2[nH]1 c1(-n2cc(CC3N(C(C4N(CC)CC4)=O)CCC3)nn2)cccc(F)n1 C(=O)(CS(=O)(=O)CC)N(n1cncn1)CC C(c1sc2ccccc2c1Cl)=CC(N1CCC(NC(C2C(C)CC=CC2)=O)C1)=O C12(C(N3CC(NC(C4C(C)(C)C4)=O)C(F)C3)=O)CC1COC21CCC1 N1(C(C2C(=C)C2C(=O)OC)=O)CCN(C(c2cc(C(C)C)no2)=O)CC1C(C)C C(=O)(C1=C(SC)CCCC1)NCC1(C)COCCN(C(C(F)=CCC)=O)C1 c1(NC(CC2CCCC(NC(C(COCC)(C)C)=O)C2)=O)ccc(CO)c(F)c1 c1(C(C(=O)NCCCN(C(C2CC(F)C(=O)N2)=O)CC)C)cc(F)cc(F)c1 c1(NC(C2CCCN(C(=O)Nc3scc(CC)n3)C2)=O)ncc(Br)c(C)n1 CCCCCCCN(C)C(c1ccsc1C(=O)O)=O c1(C(=O)NC2CCCN(C(C3CCCC(C)C3)=O)C2)cccc(Br)c1Br N1(C(Cn2nnc(C)n2)=O)CCC2CCCC12CNC(c1scnc1C)=O N1(c2n(CCOC)c(-c3cccc(=S)n3O)nn2)CC2(CCCCC2)C1 C(=O)(C(C)(C)C1CCN(C(=O)C(C)n2ccnc2)C1)NC1C(CC(C)C)C1 c1(C(N2CCC(C)(NC(C(C)OCC3CC3)=O)CC2)=O)ccc2c(c1)CCCS2 N1(C(CSCC)=O)CC(CNC(c2csc(C(F)F)c2)=O)C2(CC2)C1 CCCCC(CC)C(=O)N1CC(F)(F)CC1CNC(C12COC(COC)(C1)C2)=O Cc1[nH]c2ncnc(N3CCN(C(c4ccc(-c5ccco5)s4)=O)CC3)c2c1C C(CC(CC)(CC)NC(=O)CCNC(=O)CO)NC(c1n(CC)nc(C)c1)=O N1(C(c2cnc(C)s2)=O)CCN(C)CC1CNC(c1ccc(F)cc1)=O CCCCCCCN=c1cc[nH]cc1S(=O)(=O)NCC1C2CCCC12 CON=Cc1ccc(C(=O)NC2CN(C(C3(CO)CCOCC3)=O)C2)cc1 N1(C(CCCCCOC)=O)CCC(NC(c2cn(C)c(C)n2)=O)C(C)(C)C1 c1(C(=O)NCC2CN(C(c3n(CC)c(O)nc3)=O)C3C2C3)ccc(OC)cc1F c1(C(=O)NCC(c2ccccc2)NC(C=NOC)=O)c(Cl)nn(C)c1Cl N1(C(C2(CCOC)CC2)=O)CC2CCCC(C1)N2C(C1(OC)CCC1)=O C1(CNC(CC=C=C)=O)CN(C(=O)C(O)Cc2cc(Cl)sc2Cl)CC12CC2 C(=O)(C1=NN(C)C(=O)CC1)N1CCC2C(NC(CN(C)C(c3ccsc3)=O)=O)C21 C1(O)(CNC(C2(C)CC=CC2)=O)CCN(C(=O)CCCOc2cccc(F)c2)C1 C1(NC(C(C2CCOCC2)C)=O)CN(C(C2(C)CCOCS2)=O)CC1CO C1(O)(CC(=O)N(C(C)C(=O)NC)Cc2cccc(C(=O)NC)c2)CCN(C)CC1 C(=O)(C(C(C)CC)N1CCOCC1)N1CC(C(=O)Nc2cn(CC)nc2)OCC1 c1(C2(C(=O)NCC3(F)CN(C(C4(C)CC4F)=O)C3)CC2)ccccc1F c1(C2(NC(CCOCCNC(=O)C=Cc3ccoc3)=O)CCC2)ccnc(Cl)c1 C1(CC(=O)NCC=C(C)C)CC(C)N(C(C2CCOC2(C)C)=O)C1 c1(C(=O)OCC)cc(C)nnc1N1CC(O)(C(C)NC(=O)C(C)CC(C)C)C1 C1(C(N2CC(NC(COC)=O)C2)=O)C2CCC(C2)N1C(=O)C(N1CCNC1=O)C c1(NC(=O)Nc2scc(CCC(=O)OC(C)(C)C)n2)cc(C#N)c(F)cc1F C1(CC)CN(C(c2ccn(CC)n2)=O)CCC1NC(c1c(C)cncc1C)=O Cc1n[nH]c(C)c1C(=O)NCC=CCNC(C1CC1(C)C(F)F)=O N1(C(c2[nH]cc(CC)c2)=O)CC2(C1)CN(C(=O)COC1CCOCC1)C2 C1(NC(C(C(CC)C)OC)=O)CC2(CCC(NC(=O)CCC3CC3)CC2)C1 C1(NC(C2CC3(CCC3)C2)=O)CC2CCC(C1)N2C(C1CCOC1C1CC1)=O C1(NC(C(CCC)O)=O)CCC2CN(C(C3CNc4ccccc4C3)=O)CC2C1 N1(CCc2n(C)nnc2)CCCN(C2(C(=O)O)CC2)CC1 C(=O)(CC(C(=O)Oc1ccccc1)NC(C1CC2(CC2)CN1C(=O)C1CC1)=O)OC Cc1cc(OCc2nc(-c3cncnc3)nn2CC(F)(F)C(F)F)cc(C)c1 N1(C(C(C)C2CCC2)=O)CC2CC(NC(=O)CCc3cncs3)C1C2 C(=O)(C(C#N)C(C)C)NC(CN(C(c1cc(C)[nH]n1)=O)CC)C c1(OCCC(=O)NCC2(O)CCN(C(COCCSC)=O)C2)cc(C)cc(C)c1 c1(OC)cc(C(=O)NCC2CC(F)CN2C(=O)Cn2cnc(=N)[nH]2)c(F)c(Cl)c1 c1(C(=O)NC2CC(C)(NC(Cc3n(C)cnn3)=O)C2)cccc2nc(Cl)cn12 N1(C(c2ccc(=N)[nH]c2)=O)CC2CCC1C(NC(c1nccn3nccc13)=O)C2 N1(C(C(CC=C)(F)F)=O)CCC2(CC1)CC2NC(=O)COCc1cc(C)on1 C(=O)(C1=NN(CC)C(=O)CC1)N1CCC(N(CC#C)C(C2CC2(C)CC)=O)CC1 N1(C(C(CCC)C)=O)CC2CCN(C(=O)CN3CCCCCC3)CC2C1 CC1=C(C(=O)NC(C)CN(C(=O)C(C)(C)N2CCCCC2)C)S(=O)(=O)CCO1 N1(C(C2C(=O)NCC2)=O)CCC2C(CCCN2C(=O)CCc2cccnc2F)C1 N1(C(COCC=C)=O)CC(O)C(O)C1CNC(C1CN2CCC1CC2)=O C12(C(N(C3CN(C(C(C)CC4CCCO4)=O)C3)C)=O)CCC(CC1)C2(C)C c1(CC(=O)N(CC(C)(C)CNC(C2CCC(CF)C2)=O)CC)ccc(C#N)cc1 n1(CC)nc(C(=O)NC(C)CN(c2nc(CCOC)ns2)C)ccc1=O Cc1oc(Cl)nc1C(N1CCC(C(C(C)C)NC(=O)COCC(C)(C)C)C1)=O N1(C(c2n(C)nnc2)=O)CCC(NC(c2cnc(Cl)cc2N)=O)C(CO)C1 C=C(C)CC(C(=O)NC1(C(N2CCC2)=O)CC(F)(F)C1)OC N#Cc1ccc(N2CCC(C(N3CCC(c4nc(=O)o[nH]4)CC3)=O)CC2)nc1 Cc1ccc(C(=O)NC(C2CCCN2C(=O)Cc2csc(Br)c2)C)nn1 Cc1sncc1C(=O)NC1CC1NC(=O)C(C)N1CCC1 c1(C(=O)NCCC2CCC(NC(CN(C)CCO)=O)C2)cc(N)ccc1Br c1(CNC(c2n(CCSC)nnn2)C2(c3cccs3)CC2)cccc(F)c1C c1(C(C)C(=O)NC23CC(CNC(c4conc4C(C)C)=O)(C2)C3)ccccc1F C1(CC)CC(O)CN1C(c1ccc(OC)nc1)C(=O)NC1CCC(C(=O)OC)C1 C=C(C)CC(C(=O)N(CCC(=O)NCCCOC)C(C)C)OC C1(C(=O)NC2(C(=O)NCC3C(C)(C)C3)CCOCC2)Cc2ccccc2C1 N1(C(C(c2ccccc2)OC)=O)CCCC2(NC(=O)CC(C)(C)C)CCCC12 C(CO)(CC(C)(C)C)NC(CN(C(=O)CC1CSC1)CCC)=O c1(C(N2CCN(C(C3(C)CCN(C)C3)=O)CC2CF)=O)cccc2ccnn12 c1(C(N(CCNC(c2oc(CC)c(C)c2)=O)C2CC2)=O)cc2n(n1)CCCO2 c1(C(N2CCCC(C(C)NC(CC(CC)CC)=O)C2)=O)ccc2c(c1)COC2=O CC(C)C(C(=O)NCCCC(C)NC(c1c(N(C)C)cccc1F)=O)NC(N)=O c1(C(N2CCC3(C(=O)NC4C(C)CN(C)CC4)C(C2)C3)=O)cc2ccccc2s1 CCCC(CO)N=c1[nH]c2cc(Cl)c(S(=O)(=O)NC3(C4CCC4)CC3)cc2s1 c1(COC)cccnc1C(=O)NC12CC(CNC(C3CCCN(C)C3)=O)(C1)C2 c1(N(C)C)ccc(C(n2nc(-c3cccs3)nc2-c2cccs2)C2CC2)cc1 C1(C(=O)NCC(NOC)=O)CCCN(C(c2ccsc2OC)=O)CC1 N1(C(C2CC(C#N)(OC)C2)=O)CC(C)C(C)(CNC(=O)C(C)C2CC2)C1 N1(C(CCCN(C)C)=O)CCC2(CC1)CN(C(C1(F)CCOC1)=O)CCO2 C(CCCCC(=O)N(C)Cc1nnc(C)s1)N(C(c1c(CC)n[nH]c1)=O)C c1(N2CCC(NC(C34CCCCN3CCC4)=O)C(O)C2)ncnc2ccsc12 C(CCCCCCO)NC(CC(CNC(=O)CCC1CC1C)OC)=O c1(CCC(=O)NCCOC2CC2c2ccccc2OC(F)F)ccc(F)cc1F C=CCC(C)(CC)C(=O)N1CCC(CN(C)C(C2(C)CCN(C)C2=O)=O)CC1 C1(O)(CNC(C(C)OCCOC)=O)CCN(C(C2CN(C)C2)=O)CC1 N1(C(c2c(C)ncs2)C(=O)NCC2CCOC2)CCOc2c(Br)cccc2C1 C(=O)(C(CC(C)C)ONC(=O)C=C(C)C(C)C)NCCOC(C)=O C1(C(N2CC(C)(NC(C3CCCO3)=O)C2)=O)CCOC1(C)C C(=O)(C#CC1(C)COC1)N1C(CNC(c2cn(-c3ccc(C)cc3)nn2)=O)CC1 C(CC(C)(O)CNC(C1OCCC1CNC(=O)C(C(C)C)C1CCC1)=O)OC c1(C(=O)NC(C2CCN(C(=O)COC(F)(F)F)CC2)C)cc(F)n(C)n1 N1(C(C(CC)NC(N)=O)=O)CCN(C(=O)C(=O)NC2CC2)CC1CC(F)(F)F C(=O)(C(CC(C)(C)C)OC)NC1C2CC(NC(C(CCSC)OC)=O)CC21 Cc1ccn2c(C(N3C4CCC3C(F)C(NC(C3CCOC3)=O)C4)=O)cnc2c1 C(C)(C(C)(C)C(=O)NCC1CN(C)CCN1C)NC(c1n(CC)ncc1)=O Cc1c(NCc2cscc2-c2ccncc2-c2cccc(I)c2F)cccc1F Cc1cc(C(=O)NCCCOCCCNC(=O)COC(=O)CO)oc1C c1(COC)ccc(C(=O)NCC2C=CCN2C(=O)C(C)CO)cc1OC C1(N(C2CC(=O)N(C(C)C)C2)C(C(COC)NC(C)=O)=O)C2CCC1CNC2 N1(C(c2cccc(C)c2F)=O)CCCN(C(=O)CC2CCCC(C)O2)C(C)C1 CC(C)C(O)C(=O)NCC(C1CCN(C(=O)COC2CCCCCC2)CC1)F c1(C(N2CCN(C(C3CCCC(C)CC3)=O)C(C)C2)=O)cnc2ncnn2c1O C1(C(=O)NCC2CCN(C(c3nc(C(C)OC)oc3)=O)CC2)CC2(CCC2O)C1 c1(C(N(CC(CC)NC(C2CC(O)C2)=O)C)=O)cc2n(n1)CC(O)CO2 CCC(C)(COC)C(=O)N1CC2CC1CN2C(=O)CCC(=O)c1ccccc1 C(C)(CC(C)C(F)F)(c1nnnn1CCSC1(C)CC1)NCC(=O)OCCCC Cc1c(C(N2CCC3C(CCN3C(=O)C(C)C(C)C)C2)=O)cccc1[N+](=O)[O-] C1(Cn2cc(CC34CC(C)(C3)OC4C(=O)O)nn2)CCCN2CCCC12 S(=O)(=O)(c1cc(Cl)cs1)Nc1ccc(C)c(Br)n1 N1(C(c2c(CC)nn[nH]2)=O)CC(CNC(c2nccn2C)=O)CCC1C n1(CC)nc(C(N2CCCC(CNC(c3ccc(Cl)o3)=O)C2)=O)cc1C CCC(COC)(CC)C(=O)NCc1cc(O)cc(Br)c1.C1(=O)CO1 Cc1csc(=NCC(=O)NCCCNC(=O)C(c2ccc(C)s2)C)[nH]1 N1(C(=O)Cc2ccc(Cl)s2)CCN(C2CCC(NC(=O)C3=COCC3)CC2)CC1 c1(C(N2CC3CCN(C(CC(C)OC)=O)C3C2)=O)cccc2c1oc(=O)n2C C1(NC(C2(CC#C)CCCCO2)=O)COC2(C1)CN(C(=O)CCCC(C)(C)C)C2 N1(C(C(C)SCCCC)=O)CCCOC(CCNC(c2cnc(S)nc2)=O)C1 C12(CNC(C3(c4ccn(C)n4)CC3)=O)CN(C(C3CSCCS3)=O)CC1CCO2 CCC(CC(=O)NCC1CCN1C(C1COC(=O)C1)=O)c1ccc(C)cc1 N1(C(c2n(CC)nnc2)=O)CCC(CO)(NC(c2cc(C)n(C(C)(C)C)n2)=O)C1 Cc1cc(C(N2CCN(C(C3(C(F)F)CCCO3)=O)CC2CO)=O)cc(O)c1 C1(C(=O)NCC2N(C(Cc3c(C)ncs3)=O)CCC2C)CCC(C)(C)CC1 N1(C(C2(CC)CC2)=O)CCCCC(NC(c2ccc(OCC(F)F)cc2)=O)CC1 c1(N2CCN(C(c3ccc(C(N)=S)cc3)=O)CC2)cnc2ccccc2c1 Cc1ccc(C=CC(=O)NC(C2(O)CCN(C(c3coc(C)n3)=O)C2)C)cn1 C1(CNC(c2cc(F)ccc2O)=O)COCCN(C(C2(O)COC2)=O)C1 CC1COc2c(C(N3CC4(CNC(C5CC(O)C5)=O)CCC3CC4)=O)cccc21 C(=O)(CCC(=O)c1ccc[nH]1)NCC(C)(CNC(=O)CC1CCOC1C)OC S(=O)(=O)(c1cc(F)cc(F)c1)N1C2CC(c3n(CC)ccn3)CC1CC2 C1(C(C)C)CN(C(c2ccnn2C)=O)CCC1NC(c1ccc(N)c(Cl)c1)=O C12(CNCC(CC)(C)Cl)CCC(CC1)N(C(c1ccnnc1C)=O)C2 c1(C(N(C2C3CN(C(CSc4nc(C)[nH]n4)=O)CC32)C)=O)ccc(CO)c(F)c1 N1(Cc2n(C)ncc2Br)CCC2(CC1)CC(Nc1ncc3[nH]ccc3n1)CO2 C1(NCc2cn(CCS(C)(=O)=O)nc2)CCC2(CCOCC2)C1 N1(C(c2nc(CC)oc2)=O)CC2CC3CC2C1C3NC(C1CC1C(N)=O)=O c1(NC(NNC(C2CC3(C(OC(C)=O)CC3)C2)=O)=O)ccc(Br)c(C)c1F CCC(C)C(O)CC(=O)N1CCCC(C)(C(=O)NC(CCO)C2CCCC2)C1 C(=O)(C(C(C)C)NC=O)NCc1onc(C)n1 N1(C(C2C(=C)C2C(=O)OC)=O)CCCC(CCC(=O)N(C)CC2CCOCC2)C1 C12(C(N3C(C(=O)NCC4(OCC)CC4)C(O)CC3)=O)CCCC1C2(F)F CCC(O)C(C)C(=O)N(CC(C)(C)NC(=O)C(=C1CCCCC1)F)C CC12CC1CN(Cc1cccc(C(F)(F)C(F)(F)F)c1)C2 c1(C(=O)O)cc2c(cc1NC(C1CC1c1ccncc1Cl)=O)OC(F)(F)O2 c1(CN(C(=O)NCc2c(OC)nsc2OC)C)ccc2n[nH]cc2c1Cl c1(C(=O)Nc2cnn(Cc3ccncc3)c2)ncccc1-n1cccn1 CC1CCN(C(c2cccnc2F)=O)CC1NC(=O)CCCCCO C1(NC(Cc2cc(CC)no2)=O)CCOC(C(=O)NCCc2ccc(F)cc2)C1 N1(C(c2c(OC)n[nH]c2)=O)CCC=C(C(=O)NCC23CCCN(CC2)C3)C1 C(CC(C)(C)C(=O)N(C)CC1CC(O)C1)NC(CC(=O)OCC)=O C1(C(N(C2C(C)CCC2)C)=O)CCN(C(c2ccc3c(c2)CCC3)=O)C12CCC2 C1(C)(C(=O)NC2CC(CNC(C=C(C)C(F)F)=O)OCC2)CC2CCC1C2 c1(C(=O)NC2CN(C(C(CC)NC(N)=O)=O)CC2C)ccc2nc[nH]c2c1F C1(NC(=O)CC2CC3CCC2O3)CC2CN(C(=O)Cn3ncnn3)CC2C1 CCC(CC(=O)N1CC(CN(C(=O)C(C2CCCCC2)O)C)C1)OC C(=O)(C1=CC2(CCOCC2)C1)NC1CC(F)(CNC(C(c2cn(C)nc2)=O)=O)C1 N1(C(c2c(CC)scc2)=O)CCC12CN(C(C13COCC1C3(F)F)=O)C2 C(=O)(CC(C=C)CC)N1CCC(C(C(=O)OCC)(F)F)(C(=O)OC)C1 C1(NC(c2cc(CC(C)C)on2)=O)COC2(CCCN(C(=O)C(C)(C)CO)C2)C1 c1(C(C)C)c[nH]cc1C(=O)N(C1CCCCC1)CCNC(C12CCC(C1)C2)=O N1(N(CCCC=C)C(C)C)CCS(=O)(=O)C(COC(F)F)C1 c1(C(=O)NC2CC(C(=O)NCCc3c(C)n[nH]c3C)C2)c(C)nc2ncccn12 C1(NC(C2(CC)CCCO2)=O)CN(C(c2cc(Cl)cs2)=O)CC1C(F)F C1(C(C)NC(c2ccc(SC)s2)=O)CCCCN1C(c1cn(C2CC2)nn1)=O O=C(CCCC1CCC1)NC1(CCNC(=O)C(=O)NCC(F)(F)F)CCCC1 c1(C(=O)OC)c(NC(c2ccc(OC(F)F)cc2F)=O)cccc1Br C1(C(N2CCOC(CNC(=O)CSCC(F)(F)F)C2)=O)(OC)CCC12CCC2 c1(C(C)NC(CC(=O)OC)=O)cnc(N2CCN(C(C)=O)CC2)cc1C CC1CN(C(c2ccoc2Cl)=O)CCC1CNC(=O)Cc1cc[nH]c(=N)c1 Cc1cc(NC(=O)C(CO)NC(c2ncccc2F)=O)cc(F)c1 CC1Cc2cc(S(=O)(=O)N(Cc3ccccc3)Cc3c(F)cccc3F)ccc2O1 c1(-c2cn(C3CC(C(=O)NC4C(C)OCC4)C3)nn2)cccnc1Cl c1(C(N2CCC(CSC)C2)C(=O)NC2COC2)cccc(Cl)n1 N1(C(C2(OCC)CC2)=O)CC2CC(C1)N2C(C1CCCSC1C)=O c1(C(N)=O)cccc(CC(=O)NCc2nc(CNC(C3(C4CC4)CC3)=O)cs2)c1 N1(C(C(Cc2ccc(OC)cc2)C)=O)CCCC(CCNC(=O)C(C)(Cl)Cl)CC1 CCN(OC)C(=O)CNC(C1(N(C(=O)C(C)(C)CO)C)CC1)=O C(=O)(CCCCCCNC(C1CCCOC1)=O)NC(c1c(C)noc1C)C1CC1 C(=O)(CC(F)(F)C(C)(F)F)NCC(CN(C(CC(c1c(C)noc1C)C)=O)C)O CCC(CC(F)(F)F)C(=O)N1CCC2C(NC(c3c(C)nn(CC)c3C)=O)C12 C(C(C)(O)CC(=O)NC1(CC(N2CC(S(C)(=N)=O)C2)=O)CCC1)OC c1(N2Cc3c(nc(C)s3)C2)nc(=NC(C)c2ncc(Br)cn2)[nH]c2c1cnn2C C(=O)(C1=CCOCC1)N1CC(NC(CCC(=O)N(C(C)C)C)=O)C(F)C1 N1(C(C2ON=C(CC)C2)=O)CC2(CCCC2NC(c2c[nH]nc2C(C)(F)F)=O)C1 C1(C(CCNC(C2CCN(CCSc3ccccc3)C2)=O)O)CCOCC1 c1(C(=O)NC2CC(NC(CC(c3c(C)cccc3)C)=O)C2)ccc(Cl)c(O)c1N c1(C(=O)NC2(CNC(C(CC)n3nccc3C)=O)CCC2)cc2cnn(C)c2s1 c1(C(=O)NC2CN(C(C(C)P(C)(C)=O)=O)CC2O)nc2ncc(CCO)cn2n1 Cc1cc(C(=O)NCC2C3CN(C(=O)CN4C(C)CCC4C)CC23)oc1C C1(C(=O)NC2(C(F)F)CC(NC(=O)Cc3ccon3)C2)CCCCC(=O)N1 c1(CCC(N2C(CNC(C3CC3(F)F)=O)CCC2)=O)ccc(C(F)(F)F)cc1 C1(CC(=O)NCCC(N)=O)CN(C(C2CC2c2ccccc2)=O)CCO1 CC1CCCC(C(N2CCSCC2C(C)(C)N(C2CCOCC2)C)C(=O)NC)C1 C1(CS(C)(=O)=O)(C(=O)NC(CC)(C)CNC(=O)CCCSC)CC(F)(F)C1 N1(C(c2ccc(NC)cc2)=O)CCCC(C2CCN(C(=O)CC(F)F)CC2)CC1 C1(NC(C2C(C)CCOC2)=O)CN(C(=O)C(F)(F)C(C)(C)O)CC1C1CC1 C1(N(C(C(C)O)=O)C)CCCN(C(c2cccn(CC(F)(F)F)c2=O)=O)CC1 C1(C(N(C)CC2C(C)OCC2)=O)C2CCN(C(=O)C=Cc3ccc[nH]3)CC12 c1(NC)cnncc1C(=O)NC1COCCC1C(=O)NOC(C)C c1(OC)ncnc(OC)c1NC(C1CCCN(C(c2cccc(C)c2)=O)C1)=O N1(CC(=O)NCCC2CN(C(=O)Cn3ncnn3)CCO2)CCCNS1(=O)=O c1(OC)cccc(NC(=O)Cc2noc(CC3(C)CC(C#N)C3)n2)c1O C1(C(=O)NC(C(=O)NCC(c2ccsc2)C)c2ccco2)CC(=O)CS1 c1(OC)c(C(=O)N(CC(Cc2ccccc2)NC(C2CCCO2)=O)C)csc1C C1(C(=O)NC2(C(=O)NCC(C3CC3)C3CC3)C(C)CCC2)CCCC(=O)N1C c1(C(=O)NC2(CNC(CCc3ncc(C)[nH]3)=O)CC2)ccncc1N c1(NCCC2N(C(CS(CC)=O)=O)CCCC2C)ncc(Br)cc1[N+](=O)[O-] C1(CC(N2C(CC(=O)NCCn3cc(Br)cn3)CCC2)=O)CCCOC1 c1(CC)cc(CC(=O)NC2CC2NC(c2occc2CN(C)C)=O)on1 c1(CC)ccc([N+](=O)[O-])cc1CNC(c1cc(Br)no1)c1nnnn1C C1(CNC(C2(OC)CCOC2)=O)CC(NC(c2cccc(C(C)C)n2)=O)CCO1 C1(CC(=O)N=CC(=O)NCC2CN(C(CC)=O)C2)CCN(C)C1=O C1(C)(C(N2CCN(C(CC)C)CC2)=O)CCCN(C(c2c(C)ccn2C)=O)C1 C(=O)(C#CC1CCCO1)N1C(CCNC(c2cnc(COC)s2)=O)CCC1 C12(C(=O)NCc3c(C)nc(CC)o3)CC(CO1)N(C(C1(C(C)(C)O)CCC1)=O)C2 Cc1cc[nH]c1C(N1CCCC1C1(NC(=O)CCc2ccco2)CC1)=O N1(C(c2c(C)cns2)=O)CCC(NC(c2cc(C(F)F)nn2C)=O)C(CO)CC1 CC1(C)CC1(Cl)C(=O)NC1CCCC1NC(c1coc(C2CC2)n1)=O N1(C(C2COC2)=O)CCN(C(c2ccns2)=O)C(c2cccnc2)C1 C1(C(N2CCN(c3ncco3)CC2)=O)CCC2(CCNC2=O)CC1 C1(C)(C(N2CCCC(C(=O)OC)C2)=O)CCCN(c2ncc(Cl)cn2)C1 O=C1CCC2(C(N3CCCC(N4CCN(C(=O)C=CBr)CC4)C3)=O)CCCC2C1 CC(C)(C)C(=O)C(=O)NC1CC(NC(C2(c3cnn[nH]3)CCOC2)=O)C1 c1(NC(N2CC(Cn3cc(C(=O)O)nn3)C(C(F)(F)F)C2)=O)cc(Cl)ncc1Cl c1(OC)cc(F)c(C(=O)NCCCNC(c2cnn(C)c2C(C)C)=O)c(F)c1F CC(C)(CCl)C(=O)Nc1ccnc(C(=O)Nc2ccc(C(N)=O)s2)c1 Cc1cc(Cl)ccc1CCCNC(=O)COC(c1ccccc1Br)CC(C)C c1(C(N(CCCCN(C(=O)CCC2(C)CC2)C)C)=O)nnn2c1COCC2 c1(C(N2CC(O)CCC(NC(c3c(C)cco3)=O)C2)=O)nncc2c1CCCC2 Cc1ccc2occ(C(N3CC(C(C)NC(c4nncn4C)=O)C3)=O)c2c1 C(=O)(CCCCCC#N)NC(C(=O)NCCSCC)Cc1ccco1 CC(C)C(C)C(=O)NCC1(F)CC(CNC(c2ccc(CNS(C)(=O)=O)o2)=O)C1 c1(CC(=O)NCc2cccc(NC(C3(CF)CC3)=O)c2)ccc(F)nc1 C(=O)(CCCCCN=[N+]=[N-])NCc1c(C(=O)NC(c2ccc(C)nc2)C)scc1 N1(C(c2scc(C)c2Cl)=O)CCC(C)C(CNC(C2CNC(=O)N2)=O)C1 CC(CCC(=O)NCC1(CNC(=O)CC2OCCCO2)CCCCC1)N(C)C C1(NC(c2c(CC)ccs2)=O)CC2CCCC(C1)N2C(=O)C(C)=C1CC1 Cc1cc(C#N)ccc1C(=O)NCC(C)(C)CCNC(c1nnn2c1CCC2)=O c1(C(C(=O)O)NC(c2ccc(Cl)c(C)c2N)=O)cccc2ccccc12 c1(C(=O)NCC2COCCN2C(C2CC2F)=O)ccnc2cc(Cl)ccc12 c1(C(=O)NCC2(C(C)(C)O)CN(C(CCCC)=O)C2)cc(C(F)(F)F)nn1CC C1(O)(CCNC(CSC)=O)CCN(C(c2sccc2-n2cccc2)=O)C1 C1(NC(c2cc(N3CCCCC3)ncn2)=O)C2CN(C(=O)COCCF)CC12 c1(OC)ccnc(C(=O)NCCC23CCC2CN(C(=O)C=C(C)C(C)C)C3)c1O c1(OC)cc(C)c(C(=O)N(CC(O)CN(C)C(C2CCS(=O)(=O)C2)=O)C)c(F)c1 C(C(F)(F)F)(c1cnn(C)c1)NCC(C)COc1ccccc1 C1(CC#C)(C(N2CC(CO)(CO)C2)=O)CCN(C(C2CS(=O)C2)=O)C1 C(=O)(C#CC1(C)COC1)NC1CN(C(C(c2ccc(C)cc2)F)=O)CC1F c1(C(C)(C(=O)NCCCN(C(C2CCSC2)=O)C2CC2)OC)ccccc1F N1(c2c(C(C)=O)cccc2)CCC(NC(C2CCCCN2CC(C)C)=O)CC1C CC1(C)CC(NC(C2CCOC2(C)C)=O)CN(C(c2cn(C3CC3)cn2)=O)C1 c1(CC)cnn2ccc(C(=O)NC(C)CN(C(=O)CCC3CC3C)C)nc12 C1(C(N2C(C3CCN(C(C=NOC)=O)C3)CCC2)=O)CCC(=O)N(C)C1 CCC(C(=O)N1CC2(C)CC1(C(=O)NCC1COC(=O)N1)C2)C(C)C C1(CC(N)=O)(NC(C(CCC)O)=O)CCN(C(c2c[nH]nc2C(C)C)=O)CC1 c1(CCC(N2CC(OCC(=O)N(C)CCn3ccnc3)C2)=O)cnn(C)c1 N1(C(c2n(C)c(=O)ccc2)=O)CCC2CN(C(c3c(F)cccc3Br)=O)CCC12 c1(C(=O)NC2CCC(CCNC(c3cccc(=O)o3)=O)C2)cncc(O)c1 c1(OCC(=O)NC2CC(CNC(C3ON=C(C)C3)=O)CC2O)cccc(C)c1C c1(C(N(C2C(N(C(CCCC=C)=O)C)CCCC2)C)=O)cc(C#N)n(C)n1 C1(OC)CC(=O)N(c2cnn(CCF)c2)C1.C12(CCO)CN(C1)C2=O Cc1cc(C)c(C)c(C(=O)NC2CN(C(=O)C3=NOC(C)(C)C3)CC2O)c1C N1(C(c2ncn(C(C)C)n2)=O)CCN(Cc2ccc(Cl)c(F)c2)CC1C CCC(C(=O)NCC(O)CNC(=O)C(C#N)=CC1CC1)n1ccnc1 CCCC(CNC(c1ncc(F)cc1F)=O)C(=O)Nc1cn(CC)nc1C#N O=C(O)C#CC(=O)Nc1ccc(-c2ccc(-c3cc[nH]n3)cc2)cc1 C1(NC(c2c(OC)ccnc2)=O)CCC2CCN(C(=O)CSc3nncs3)C1C2 c1(OC)c(C(=O)NCC2CN(C(=O)C(C)(C)C)CCC2(F)F)cc(F)cc1F c1(C2C(NC(C3CC(NC(=O)OC(C)(C)C)C3)=O)CCC2)cc2n(c1)CCOC2 c1(C(=O)NC2CC23CC(NC(C2CCCS(=O)(=O)C2)=O)C3)n[nH]c2c1COCC2 c1(C(N2CC3C(NC(C(C)(CO)OC)=O)(C3)C2)=O)cccc(Cl)c1F N1(C(c2c(C#C)c[nH]n2)=O)CCC(CO)C(NC(C2(N(C)C)CCCOC2)=O)C1 C12(NCC(=O)NC3CN(C(C4(C)CCOC4)Cc4nc[nH]n4)C3)CCC(CC1)CC2 N1(C(=O)Nc2nc(CN3CCCC3)cs2)CC2OCOC2C1 N1(C(=O)C=Cc2cn[nH]c2)CC2CCN(C(c3ccc(Cl)c(Cl)c3)=O)CC2C1 N1(C(c2n[nH]c(C)c2C)=O)CC(C(=O)NCCC(C)(C)O)C(C2CC2)C1 c1(C(C(=O)N(CCNC(CC2(C=C)CCC2)=O)CCOCCO)C)cc(C)oc1C c1(C(N(CCCNC(=O)Cc2cc[nH]c2)C(C)C)=O)cccc2c1OC(C)C2 C1(CNC(C=CCN(C(c2cc(C(C)C)no2)=O)C)=O)CCCC12CC2 C1(NC(C2CC(C)(C)OCC2)=O)CN(C(=O)C#CC2CC2)CCC1(C)C c12cncc(c1)C(=O)NC2.C1(C(N2CCCCC2)=O)CCCN(Cc2ccno2)C1 C=CCC(C(=O)N(C)CCNC(C1(n2cccn2)CC1)=O)C(C)(C)C N1(C(C2CC2F)=O)CC2CC1CN2c1ccnc(N2CCCC2)n1 N1(CCC(=O)OC)CC(CN(CCC(C(C)(C)C)C(C)C)C)CC(C)(C)C1 C=CC1OCCCC1C(=O)NCC1CC1CNC(c1cc(C(C)(C)C)oc1C)=O N1(C(CCOCC#C)=O)CCN(C2CN(C(=O)C(O)C(F)F)C2)CC1 CN1CCCN(C(=O)CCCCN(C)C(C2CCC(=O)N(C)C2)=O)CCC1 Cc1cn2ccnc(C(=O)NC3CC(CNC(=O)CCCC#N)C3)c2n1 Cc1ncc(C(N2CC(O)(CN(C)C(C3CC(N(C)C)C3)=O)C2)=O)cn1 N1(C(Cc2cc(COC)on2)=O)CC(C)C(C)(CNC(c2c(C)ccn2C)=O)C1 C1(CNC(=O)CC2CCN(C3CC3)C2)(Nc2n[nH]cc2F)CCCCCC1 Cc1cccc(CC(=O)NC2CCN(C(c3cn(C(C)C)cn3)=O)C2)c1 N1(C(c2nccc(OC)c2)=O)CCC(NC(=O)CC2CCC(=O)N2C)C1(C)C c1(C(=O)NCC2N(c3ncc(C(=O)OC)c(C)c3)CCC2)cc(F)cc2ccoc12 C1(F)(C(N2CCC(OC)(CNC(c3cccc(SC)c3)=O)C2)=O)CCCN(C)C1 Cc1c(CN2CCCC2CC(N2CCC(N(C)C)C2)=O)nc2ccccn12 c1(CC(=O)NC2CCN(C(CC3C=NN(C)C3=O)=O)CC2)ccc(Br)c(F)c1 C1(C(=O)NCC(CN(C(=O)CSCc2ccncc2)C)O)CCC2(COC2)OC1 C1(C(=O)NC2CN(C(C3CCC3)=O)C3(CCC3)C2)COc2ccccc2O1 c1(N2CC3C(C(N4CCCC(C(N)=O)CC4)=O)C3C2)ncnn2c(Br)ccc12 C(C(C(=O)N(CC(C)C(=O)NC1CC(CO)C1)C)N(C)C)OC c1(C(N2CC(O)(C(C)NC(=O)Cn3cncn3)C2)=O)cccc2sncc12 n1(CC(=O)NC2(COC)CCN(C(=O)Cc3cccs3)C2)nc(C)n(C)c1=O CC(Cc1ccccc1)C(=O)NCCNC(=O)CC12CC(C1)C2 c1(CC)cc(C(=O)NCC(CNC(=O)Cc2scnc2C)OC)sc1C Cn1cnc(C(=O)NCC2CC(O)(CNC(c3cnc4n3CCC4)=O)C2)cc1=O c1(C(=O)NCCCCNC(c2ncoc2C2CCCO2)=O)ccccc1Br C1(C(=O)NC(CC=C)CNC(=O)CCCn2ccnc2)(OC)CCOCC1 c1(C(N(CCCNC(=O)CC2CCCN(C)C2)CC)=O)cnc2ncc(Cl)cn12 N1(C(C=Cc2ncn(C)c2)=O)CC2(CCN(CC3CCCO3)C2)C1 CC1COCCC1N=c1[nH]c2cc(Cl)c(S(=O)(=O)NCC3CCC3)cc2s1 Cc1cc(C(=O)NC(C)CN(C(=O)C(C(C)C)c2ccncc2)C)c(O)c(C)c1 CCC(C)CCCC(=O)NCC(C)(C)CN(C(=O)C(O)C1CCC1)C C(=O)(C1=C(C#N)CCC1)NC1CN(C(C2(OC)CCSC2)=O)CC1(C)C N1(C(C(CC)c2cccnc2)=O)CCN(C(c2ncc(F)cc2N)=O)CC1COC C1(C(=O)Nc2ccc(SC)cc2)COCCN(Cc2cn(C)nc2C)C1 N1(C(COCCCCC)=O)CC(NC(C2CCC(C(N)=O)O2)=O)C(O)C1 Cc1cc(CNC(C2(CNC(C3CC(F)(CF)C3)=O)CC3(CC3)C2)=O)oc1C N1(C(c2c(OC)nsc2OC)=O)CCC(NC(=O)C(F)n2cccn2)C(C)(C)C1 C(=O)(C(O)CC1CC1)NCCC(C)N(C(COCC=C)=O)C CC1C(NC(=O)C(C(C)O)N(C)C)CCN1C(=O)CCC1CNC(=O)N1 C#Cc1cc(C(N2CCCCC2CCN(C(=O)C(C=C)OC)C)=O)ccc1C c1(C(N(CCCNC(C(CSC)C)=O)C(C)C)=O)ccn(CCO)c1C c1(NCC(CCSC)OC)ccc(S(=O)(=O)NCCc2cnccn2)c(Br)c1 C=CCC(CC(C)C)C(=O)NCC1CC(O)CN1C(c1ccn(CC)c(=O)c1)=O C1(C)(CNC(C(N2CCC(C)C2)=O)=O)CCCN(Cc2nncs2)C1 c1(NC)ccccc1C(=O)NC(CNC(=O)CC(c1ccc(N)cc1)C)C(C)C c1(C(N2CCN(c3ncc(C)c(O)n3)C(C)CC2)=O)ccc2nc(C)sc2c1 C1(NC(C2C(CNC(Cc3nc(C)sc3)=O)OCC2)=O)CNC(=O)C1(C)C C1(C(=O)NCC2C(NC(CCOCCC)=O)C2)(OC)CCCCCC1 c1(CN2C(C(=O)Nc3c(C)ncnc3)CC3(CC3)C2)cc2ccccc2cn1 N1(n2nnnc2Br)CC2CCCC(C2)C1.N1(c2ccccn2)CCCCC1 N1(C(CSCC)=O)CC(NC(=O)CCC2C(=O)ON=C2C)C(S(C)(=O)=O)C1 N1(C(CCN(CCCCC)C)=O)CCN(C(=O)CN2CC3CC3C2)C(CCO)C1 C=CCC(C(=O)NCC1CCCCN(C(c2cncc(N)c2)=O)CC1)C(C)C C1(C(=O)NC(CC)(C)COC)COCCN(C(c2ccc(Cl)s2)=O)C1 C1(C2(O)CCN(C(=O)COCC(=O)NC)CC2)(NC(c2c(CC)ocn2)=O)CC1 c1(CCC(=O)N(C2CCN(C(c3ns[nH]c3=O)=O)C2)CCC)ccc(CC)cc1 c1(NC(c2c(NC(c3ccn(C)c3)=O)cccc2F)=O)cc(C(=O)O)ccc1C#N S(=O)(=O)(c1cnccc1N1CCCC(N)C1)N(C)N(CCC(F)(F)F)C.C(N)=O CCC(C)C(C(=O)NCc1occc1C)N(C(=O)C(C(C)OC)N(C)C)C N1(C(c2cc(CNC(C(C)n3cccc3)=O)[nH]n2)=O)CC2CCCC(O)C2C1 Cc1cc(C)c(C)c(S(=O)(=O)N2CCN(C(=O)CNC(=N)N)C(C)C2C)c1C N1(C(C2(CC#C)CCN(C(c3scnc3C)=O)C2)=O)CCCOC(C)(C)C1 C12(C(=O)NCc3scc(CNC(C4CCC(C)O4)=O)n3)CCC(CC1)CO2 Cc1cccc(C)c1CC(=O)NC(CO)C(C)NC(C1(F)CC2(CCC2)C1)=O C12(CNC(CCN3CCC(C)CC3)=O)CCC(NC(C3CC=CC3)=O)(CC1)CO2 C1(N(C)C(C2CCCN2C(c2cccc(Cl)c2)=O)=O)CC2(CCC2)C1 Cc1cc(C)c(C(=O)NCC23CCC2CN(C(C2CC2(C)C)=O)C3)cc1N C1(C)(C(N2CC(C)(OCC(=O)NCC(CC)(C)OC)C2)=O)CCN(C)C1 N1(C(=O)C=Cc2cccc(O)c2)CC(NC(C2CC(F)C2)=O)CC12CCOC2 N1(C(C(CC)O)=O)CCC(O)(CNC(C2CCCSC2)=O)CC1 N1(C(c2cc(CC)n(CCO)n2)=O)CCC2CN(C(C3(C)CSC3)=O)CC2CC1 N1(C(C(C(C)O)(F)F)=O)CCC2(COC(CNC(c3ccco3)=O)C2)C1 c12ccc(o1)CNC(=O)C(C)N(CCC)C2=O.C(=O)(CO)NCCN(C)C n1(C(C)C(=O)NC2(C3CCCCN3C(=O)CCF)CC2)cnc2ccccc12 c1(C(N2CCC(CN(C(C3C(C(=O)OC)C3)=O)C)C2)=O)cc2ccc(Cl)cc2s1 CC1(C)COC(C(=O)NCC(C2CCCC2)NC(=O)C=Cc2ccccc2)C1 c1(OC)ccc(CN2CCN(C(c3cc(Br)cnc3C)=O)CC2C)nc1Br C12(NC(C3CC(=O)N(O)C3)=O)CC(C1)N(C(c1ccccc1O)=O)C2 N1(C(Cc2n(C)cnc2)=O)CCN(C(c2cc3c(ccn3C)[nH]2)=O)CC12CCC2 c1(C(N2CCC(NC(=O)Cc3cc[nH]n3)(CF)C2)=O)nccc(Br)c1O Cc1cc(C(=O)NC2CC3(C2)CC3NC(c2[nH]c(O)nc2C)=O)nc(C)n1 N1(C(COCCOC)=O)CCCCC(CNC(C2(C(C)C)CCC2)=O)C1 C1(CNC(COCC)=O)CCCN(C(c2n[nH]cc2F)=O)C1 N1(C(C(C)NC(=O)NC)=O)CCCCC1C1CCCN1C(C1CCCC(F)C1)=O C12(CNC(CC3(CSC)CC3)=O)CCCCC1N(C(c1cncc(Cl)n1)=O)CC2 Cc1csc2ncc(C(=O)NCC3CC(C)N(C(=O)CCCCC(N)=O)C3)n12 C1(NC(c2c(C)nc[nH]2)=O)C2CCCN(CCC3CC3(Cl)Cl)C2C1(C)C C(=O)(CC1=CCCCC1)N1CC(C(=O)NCC(C)CC2CCC2)C(F)(F)C1 CCC(CC(=O)NC1CCC1CNC(C1(c2ccccc2C)CC1)=O)C(C)(C)C c1(C(=O)NC(C2CCN(C(c3cn(C)cn3)=O)C2)C)cccc2cnsc12 C(N=c1[nH]c(N2CCn3nc(CO)cc3C2)nc2c1CCC2)C1(CCC)CC1 N1(C(C(C)NC(C)(C)C)=O)CC(C(N)=O)(NC(=O)CC2CCC(C(F)(F)F)O2)C1 C1(NC(c2cccc3c2CCN3)=O)CCN(C(C2CCCCO2)=O)C12CCCC2 c1(C(N2CC(NC(c3coc(Br)c3)=O)C2)=O)cc(=O)c2cc(Cl)ccc2o1 CC1=C(C)CN(C(=O)CN2CCN(C(=O)C=CCN3CCCC3)CC2)CC1 CC(CC(N)=O)C(=O)NC1CCC(NC(=O)CCCc2cccs2)CC1 c1(C(=O)NCC(CCOC)NC(c2coc(C)c2)=O)cnc(OC)c(C)c1 C12(C(=O)NCC3(O)CN(C(CCCC(N)=O)=O)C3)CCCC(C1)C(=O)N2 c1(NCCC(C)NC(CC2(OC)CCCC2)=O)nc(Cl)nc2c1cnn2C c1(CN2CC(CC(N3CCC(OCC)C3)=O)C2)ccc(OC(F)(F)Cl)cc1 c1(C(N2CCC(C(N3C(C=C)COCC3)=O)(OC)C2)=O)ccc(C#N)c(C)n1 c1(C(=O)NCC(C(=O)NCC2C(OCC)CC2)O)n[nH]c(C)c1Cl C=C(Cl)CCC(=O)NC1CCOCC1C(=O)NC(C)C(=O)NC1CC1 Cc1nn(CC(F)F)cc1C(=O)NC(C)CN(C)C(C1CCC=CCC1)=O C1(CCNC(C=CCCC(C)C)=O)CC2CCC(C1)N2C(c1csc(F)c1)=O C1(C(N(CCCC=C)C)=O)CN(C(=O)CC(CC)C2CC2)CCN1C N1(C(CCc2ccn(C)c2)=O)CCN(Cc2cn(Cc3cccnc3)nn2)CC1 c1(C(N2CCC(CN(C)C(c3cnco3)=O)C2)=O)c[nH]c2cc(F)c(F)cc12 C(CC(C)C)(C(=O)NC1CCOC(C)(C)C1)N(C(CC1ON=C(C)C1)=O)C C1(CN)C(NC(=O)CC2CCCN2C(=O)OC(C)(C)C)C2CCCCC12 C1(C(=O)NC2(C)CN(C(=O)CCc3cc[nH]n3)C2)CC12CCCOC2 C(CCCCC(=O)NCCOc1ccccc1NC(=O)C(=O)NC)NC C1(CNC(c2nc(CC)oc2C)=O)CN(C(=O)CCN(C)CC)C(C)(C)C1 C1(c2cn(C3CC(OC)C3)nn2)CCCCN(C(=O)CN2CCC(C)(C)CC2)C1 c1(C(=O)N(C2CCNC2)C2CC2)c(F)ccc2[nH]ccc12 CC1(C(=O)NCC2CCCN2C(=O)CSS(C)(=O)=O)CC=CCC1 C(=O)(C1CCCc2ncccc21)NC(CC)CNC(=O)C=C(C)c1cccs1 N1(C(C2N(C)CC(C)(C)C2)=O)CC(C)(C)CCC1CNC(c1cn(C)nn1)=O c1(C(=O)NCC(N(C(C(C)CC(F)F)=O)C)C2CC2)[nH]cc2c(=O)n(C)ccc12 CCCCC(F)(F)C(=O)NCC1CCCCN(C(=O)CC2CCOC2(C)C)C1 c1(C(=O)OC)nn(C)c(C)c1CNC(=O)NCCc1cccnc1Cl C(CCN=C(NCC(=O)NC1CCC1)N1CCC(C)(c2cccc(F)c2)C1)SC N1(C2CCC(N(C)C)CC2)C(=O)NC(Cc2ccccc2)C1=O CCC(C)CCCC(=O)NCC(CC(=O)NC1CC1(C)C)OC C12(C(=O)NCc3oc(C)c(C(=O)NC(C)C(=O)NC4CC4)n3)CCC(F)(CC1)C2 c1(CC)cccc(C(=O)NC(Cc2cn[nH]c2)C(=O)N2CC(C(=O)OC)C2)c1 O=C(C(O)C(F)(F)F)NC1CC2CCC1N2C(=O)Cc1cc(Cl)sc1Cl Cc1nc(NC(CNC(=O)C=Cc2cn(C)nn2)C(C)C(C)C)cc(C#N)n1 c1(CNC(CCOCCCNC(c2cn(CCOC)nn2)=O)=O)cc(C)ncn1 Cc1ccc(CC(N)CC(=O)NC(c2c(C)noc2C)C)cc1 Cc1nc(C(=O)NCC(C)NC(C2OC(C)CC2C)=O)c2ccnc-2[nH]1 N1(C(c2nc(C(C)OC)oc2)=O)CC2C(CNC(=O)CCSC)C2C1 Cc1nc(S)sc1CC(=O)NC1CCCN(C(=O)CCc2nc(C)c(C)o2)C1 Cc1nn(C)c(NCC2CCN(Cc3cnc(C(C)C)s3)CC2)c1C=O C1(CC(=O)NC2CN(C(C3(COC)C=CCC3)=O)CC2SC)CCC(F)(F)CC1 c1(CN2C(C(=O)Nc3ccc(CC)nc3)CC(F)C2)ccc(Cl)cc1F C1(NC(Cn2c(C)nnn2)=O)CC2CCC1N2C(=O)CCCC(=O)c1ccccc1 C(=O)(C(O)C(C)(C)C)N(C)CC1CCN(C(C2CC(=O)C2)=O)C1 N1(CC(=O)N(C2CC3C=CC2C3)C(C)=O)CC(N2CCOCC2)CC1=O c1(C(N2CCCC(NC(C(CSC)O)=O)CC2)=O)cccc(S(=O)(=O)N(C)C)c1 c1(NC(N(CC)Cc2ccccc2)=O)cc(Cl)ccc1ON1CCCC(O)CC1 CC(CCCNC(c1ncc(C(F)(F)F)s1)=O)NC(c1ccsc1C(F)F)=O c1(C(=O)NCC=CCNC(C2(C)CCCNC2=O)=O)cccc2ccncc12 CC(CC#N)C(=O)NCCCN(C)C(C1CCCCN1C)=O CC(C)C1=NOC(C)(C(=O)NCC2CN(C(=O)C3=CCCCO3)CC23CCC3)C1 N1(c2snc(COC)n2)CCCCC(CNC(c2ccc(OC)c(O)c2)=O)C1 N1(C(=O)OC(C)(C)C)CC2CC(NC3CC34CCCCC4)CC1C2 C1(NC(C(c2cnn(C)c2)C)=O)CC1C1CCCN(C(=O)Cc2cnnn2C)C1 C(CC(C(=O)NCCc1ccns1)NC(c1ccn(C(C)C)n1)=O)OCC C1(C(=O)NCC(C)(C)C(N)=O)C2CC3C1C3C2N c1(C(=O)NCC(CC)NC(=O)COCCN(C)C)ccc2c(c1F)CCC2 c1(C(=O)NC(CC=C)CNC(=O)CC(C)CN(C)C)ccc(-n2cncn2)cn1 C1(C(N2C(CCNC(C=CCN(CC#C)C)=O)CCC2)=O)CC(=O)NC(C)C1 C(=O)(C(C)CC(C)(F)F)N1CCC(CNC(N2CCCC(OC)C2)=O)CC1 c1(C(=O)NCCN(C(c2sccc2Cl)=O)C2CC2)cncc2n[nH]cc12 c1(C(N(CCCN(C(C(CC)CO)=O)C)C)=O)coc(S(C)(=O)=O)c1 N1(C(C(n2c(C)cc(C)n2)C)=O)CCCN(CCNC(=O)C(C)C2CC2)CC1 C12(NC(C3(COCC)CC3)=O)CCCN(C(c3cncn3C)=O)CC1C2 c1(NC(C(c2c(Br)cnn2C)N(C)CC2CCC2)=O)ccc(Cl)cc1F c1(C(N(C2CN(C(=O)Cc3cn(C)nn3)CC2(C)C)C)=O)nc2c(s1)CCCC2 C1(COC)(CNC(c2cccs2)=O)CN(C(C2CCN(c3ncccn3)C2)=O)C1 C(=O)(C#CC1CCOC1)N1CCCCC(CCC(=O)NC2CC(C)(C)OC2=O)C1 Cc1cc(C(F)(F)C(=O)NC(CNC(c2c[nH]nc2C(C)C)=O)CO)cs1 N1(C(c2cn(CCC)nn2)=O)CC(C(=O)NCCCN2CCC2)C(C)C1 C(C(C)NC(=O)C(c1ccccc1)OC)(C(C)C)NC(CCn1nc(C)nc1)=O N1(C(C2(CCC)CCC2)=O)CC2CN(C(=O)C3=NOCC3)CC2(C(F)(F)F)C1 N1(C(C(C(C)C)NC(C)=O)=O)CC2CC1CC2CNC(c1nccc(N)c1Cl)=O Cc1c(-c2cn(CCC(=O)NC(CCO)C3CCC3)nn2)cccc1Br O=S(=O)(c1ccc(NCc2cnsc2)c(Br)c1)NCC1COc2ccccc2O1 Cc1c(CCC(N2CCOC(CN(C(=O)Cc3ccsc3)C)C2)=O)cnn1C c1(CCC(N2C(C(=O)NCC(=O)OC)CSC2C)=O)c(C)nc2ncnn2c1C c1(NCc2ccc(SC(F)F)cc2)nccc(=NCCn2cc(Br)nn2)[nH]1 Cc1cncc(CC(=O)NCC2(C(C)(C)C)CCN(C(=O)C=CS(C)=O)C2)n1 C(=O)(CCN(OC)C(=O)c1c(C)nn(C)c1C)N1CCC(NC(=O)OC)CC1 CC1(C(=O)NCCC2CN(C(=O)COc3cccnc3)C2)COCCO1 N1(C(c2c(CC)cccc2)=O)CC2(CCC2)CC1CN(C)C(C)C N12CCC(C1(C)C)CNC2=O.C(=O)(C(=O)NCC1CC1)NCC(=O)OCC c1(C(=O)NCC(C)(C)NC(c2cc(C)oc2)=O)c(Cl)ccc2ccncc12 c1(C(=O)NCC(C)NC(c2ccn(CCC)n2)=O)c(OC)cnc2ccccc12 N1(C(C=CCCC)=O)CC2CN(C(C3CCN(CC)C3)=O)CC2C1 CCCCCC(C)CC(=O)N1CCC(C)(C(=O)N(C)CC2CCOC2)CC1 CCC(O)CN(C(=O)COCCNC(=O)COCCC)CC C(=O)(C1CCCc2ncnn21)NCC(n1cc(CN2CCN(C)CC2)nn1)C C1(C(C(=O)OC)N(C(C(=O)NC(C)(C)C)c2ccsc2)C)CCOCC1 C#Cc1cccc(C(=O)NC2CC(C(=O)N(C3CC3C3CC3)C)C23CCC3)c1 c1(C(N2CC(CC(C)NC(C(n3c(C)ccn3)C)=O)C2)=O)ncc(N)cc1Cl C1(NC(C2CC(C)(CC)C2)=O)CC2CC(C1)N(C(=O)CC1CC(OC)C1)C2 C(=O)(C(O)C(C)C)N(C1CCS(=O)(=O)C1)CC=C N1(CCCNC(CC2(CC=C)CCCC2)=O)CCN(C(C2(C)CC2(F)Cl)=O)CC1 C=CCC(C)(C)C(=O)N1CC2(CCC2NC(c2cn3ccsc3n2)=O)C1 C(CO)(C(=O)NC1CC1NC(=O)CNC(=O)CSc1ccccc1)N(C)C CC(O)CCCCCC(=O)NCC1CN(C)CCN1C(c1ccc(N)cc1Cl)=O C1(C(=O)NCC2CC(OCC)C2)CCN(C(=O)C2CC3CC2CC3O)O1 N1(C(CC(C)OC)=O)CCCC12CCN(C(=O)C(c1ccccc1Cl)(F)F)C2 C1(C(N2CC(C)C(N(C(=O)Cn3cncn3)C)CC2)=O)CCC(N=[N+]=[N-])CC1 CN1CCc2c(C(=O)NC34CC(Nc5ncnc6[nH]ccc56)(C3)C4)cccc21 C1(C(=O)Nc2cccnc2Cl)CCCN(C(=O)COC2CCCCC2)C1 N1(C(c2n(C=C)nnc2)=O)CC(NC(c2cnccn2)=O)C(C2CC2)C1 C#CC1(C(=O)NC(c2ccc(C)nc2)C)CCN(C(c2[nH]nnc2CC)=O)C1 c1(C(=O)NCC(CNC(c2n(CC)nnc2)=O)O)cc(C2CC2)ncn1 Cc1ncc(Br)c(C(=O)N(C(C)CCNC(=O)C(F)=CC2CC2)C)n1 C(=O)(CCC(=O)N1CC(CNC(c2cccnc2)=O)C(O)C1)N(C)C N(C1CCCc2c(Br)cccc21)C(C(N1CC=C(C)CC1)=O)=O C1(C(=O)NC(CN(C)C)CO)CN(C(C2CC2Cl)=O)CCN1C C1(NC(C(N2CCC(C)C2)=O)=O)CCC(C)(NC(c2ccoc2C2CC2)=O)CC1 c1(OC)ccc(Cl)c(C(=O)NC2CCCC(NC(c3cc(C)nn3C)=O)C2)c1N N1(C(=O)NCCC#C)CC2CCN(C(c3cc(C(=O)OC)cs3)=O)C(C2)C1 c1(C(=O)NC2(CNC(c3cccc(CC)c3C)=O)CC2)cc2ccccc2[nH]1 C12(C(N3CCCC(NC(C4(C(N)=O)CCC4)=O)C3)=O)CCOC1CC(=O)NC2 C12(C(=O)NC3(C=C)CC3)CCC(CC1)N(C(c1nn(C)cc1Cl)=O)C2 CCC(CC(F)F)C(=O)N1CCCCC1CNC(C1CC2(C1)CC(O)C2)=O C(=O)(C(C)(C)C1=CCSCC1)NC1C(SC)CN(C(C23CC(F)C2C3)=O)C1 c1(CCCNC(=O)NC2CN(C(C(C)=CC)=O)C2)ccccc1 N1(C(C2OCCN(C(=O)CC3(O)CCCOC3)C2)=O)CCCC(F)(F)CC1 N1(C(C=CC(CC)C)=O)CCC2C(NC(=O)Cn3nnnc3C)CC12 N1(C(c2n(C)ccn2)=O)CC2CCC(NC(=O)C(F)Cc3ccccc3)CC2C1 c1(OC)cc(C(N2CCCCC(NC(c3sccc3Cl)=O)C2)=O)c(Cl)cn1 C(=O)(CC1=NN(c2ccccc2)C(=O)C1)N1CCC(O)(CNC(C)=O)CC1 c1(C(N2CCC(C)(CNC(COCC(=O)OC)=O)C2)=O)sc2nccn2c1C c1(CC2N(C(C3CCCN(C(=O)NCC)C3)=O)CCCC2)ccc(C#N)cc1 c1(C(=O)NC2C(CNC(CC(C)CF)=O)CC2)cc2cccc(Br)n2c1 C(C(=O)NCCCOCCCNC(c1cn(C)nc1O)=O)(C(C)(C)C)OC N1(CC)CCC(CNC(=O)CCC2CN(C(=O)CCCOC(C)=O)C2)CC1C C1(NC(c2cnc(OCC)s2)=O)CCN(C(=O)CCCc2cccnc2)CC1O C1(NC(C2N(C(C(C)Cn3cccn3)=O)CC2)=O)C2CCCCCC12 N1(C(C=C(C)C)=O)CC2(CCNC(c3cccc(O)n3)=O)CCC1CC2 C1(C(N2C3CC(NC(C(CCC)C)=O)(C3)C2)=O)CN2CCCN1CC2 c1(COC)nc(OC)cc(N2CC(NC(C3(C)CC(C)=NO3)=O)C(C)(C)C2)n1 c1(C(N2C(C(C)(C)NC(CNC(CC)=O)=O)CCC2)=O)cc(C)cnc1OCC c1(C(N(C)CCOCCNC(c2ccc(Cl)cn2)=O)=O)c[nH]cc(Br)c1=N N1(C(c2n(CC)ccn2)=O)CC2(CCN(C(C3CSC(C)=N3)=O)CC2)C1C(C)C S(=O)(=O)(c1cccc(F)c1)NCC(N1CCC(CNC(CCCOC)=O)C1)=O C1(C)(C(=O)NCC(CC=C)O)CC12CCN(CCCCCF)CC2 c1(C(=O)NCC2N(C(C(N3C(=O)CCC3=O)CC)=O)CC2)c(F)ccc(Cl)c1N N1(C(CC(C)(C)SC)=O)CC(CNC(C2CC(F)(F)CS2)=O)CC1(C)C Cc1ccc2c(C(N3CCOCC3CCNC(=O)C(F)C(F)(F)F)=O)coc2c1 C1(C(N2CC(CNC(C3CC(C(C)C)C3)=O)(OC)C2)=O)(OC)CCSC1 C(C)(C(=O)NC(C(=O)N(C1CC1C)C)c1cccs1)OCC c1(C(=O)NC2CN(C(c3c(CC)con3)=O)CC2C)noc2ncccc12 c1(N2CC=CC(NC(c3nc(C(C)C)oc3)=O)C2)ncn(C)c(=O)c1Br C(=O)(C(C)(O)CNC(=O)CC(C1CC1)NC(c1ccoc1C(C)C)=O)OC CCCCC(C(=O)NC(C)(C)CCCC(=O)NC(c1cccc(C)n1)C)C(C)C CCCC(CC(C)C)C(=O)NC(CCN(C)C(c1cc2n(n1)CCC2)=O)C(C)C C1(c2nnc(C)o2)CN(C(C2CN(C(C)C)C2)=O)CCO1 C1(COC)(NC(=O)Cc2nccn2C)CCN(C(=O)CC2CCSCC2)C1 C1(CCNC(C=C(COC)C)=O)CN(C(c2cnc(Cl)n2C)=O)CCO1 C1(NC(C(c2ccccc2Cl)C)=O)CCCC(N=c2[nH]c(Cl)nc3c2CCC3)C1 N1(C(C(C2CCC2)NC(C(C)=CC2CC2)=O)=O)CCOC2CC12 C(=O)(C1=COCCO1)NC1CCCN(C(Cn2c(CCC)ncc2)=O)C1 N(C(=NCCCN1CC=CC1)NC1CCOC(C2CC2)C1)CCCSC Cc1cnc(C(N2CCCN(C(c3ccccc3SCCO)=O)CC2)=O)cc1Cl c1(OC)cc(C(C(=O)NC2CC(F)(F)C2)N(CCCOC(C)C)C)ccn1 c1(C(=O)NCCCCC(C)NC(C(CC)O)=O)cc(F)ccc1N Cc1c(Br)c(C(N2CC(C3(NC(c4cnc(S)nc4)=O)CC3)C2)=O)nn1C c1(C(=O)NCC2CC(O)CN2C(c2cccnn2)=O)c[nH]c2ccc(F)cc12 N12CC(OC(C)C1)Cc1n(CC#C)c2nn1.c1(CN(C)C)ccccc1 c1(N(C)Cc2cn(CC)nc2)ncnc(NCc2cc(F)ccc2Br)c1C N1(CC(C)(C)O)CCCC1CNC(=O)NCC1(c2ccccc2)CC1 C(C(C(C)C)NC(=O)CC1CCCN1C(=O)COc1ccccc1)OC C12(CNC(c3ccc(-c4cn(C)nc4)o3)=O)CC(CO1)N(C(=O)C1=CCC1)C2 C(=O)(C(C(C)C)C1CCC1)NCC(C(=O)NCCCn1c(C)nnc1)C c1(COC)cc(NC(C2CC2(C)Br)=O)ncn1 Cc1cc(O)nc(C)c1C(=O)NCCCCCCNC(=O)CSC1CCCCO1 c1(OCC(=O)NC2C(C)CN(C(=O)CCc3nncs3)C2)ccc(F)cc1O c1(OC)c(C2CCN(C(=O)NCC3CCCSC3)CC2)cnn1C c1(C(N2C(CNC(c3cccc(Cl)c3)=O)CC(OC)C2)=O)cccc(S(C)=O)c1 C1(CN(C(C2CCC(C(C)C)C2)=O)CC)CCCN(C(c2cc(Cl)cnn2)=O)C1 C#Cc1ccc(CCC(N2CCCC(NC(c3cnc(O)n3C)=O)C2C)=O)cc1 C(N1CCN(CCc2ccc(F)cc2)CC1)n1ncc(C)c1Br S(=O)(=O)(c1ccc(N2CCc3c(Cl)cccc3C2)nc1)NC(C)(C)CC1CCC1 C1(C(=O)NC23CCC(C2)C3)CCCN(C(=O)C(c2ccccc2)F)C1 C(=O)(C(F)C(F)(F)C(F)(F)F)NC1(C)CC(NC(CCC(=O)OC)=O)C1 CC1CC(CNC(c2coc(C(F)(F)F)c2)=O)CN1C(=O)CCN1CCOC1=O C(=O)(CC(F)(F)F)N1C(C2(NC(CC3ON=C(C)C3)=O)CC2)CCC1 C1(CC(N2CC(C)C2(C)C)=O)N(C(=O)Cc2ccon2)CCC1(C)C N1(C(C(C(CC)C)=O)=O)CC2CCN(C(=O)CC3(COC)CC3)C2C1 C(=O)(C#CC1CCCOC1)NCC1(NC(C2CC(C(F)F)(OC)C2)=O)CC1 c1(C(N(CC(C)CNC(=O)CCc2ccoc2)C)=O)ncn2c1CCCC2 C1(CNC(CC2CCC(OC)CC2)=O)C(C)CCCN1C(C1CC12CC(O)C2)=O C1(C(=O)NCC23N(C(CCCC#N)=O)C(CC2)CC3)CCc2ncnn2C1 C1(NC(C(CC=C)C)=O)CCC2(CCN(C(=O)CN3CCCC3=O)CC2)C1 C1(NC(c2n(CC)ncn2)=O)CN(C(c2n[nH]c(C)c2Br)=O)CC1O C1(NC(C(CCC)OCC)=O)CCCN(C(c2[nH]cc3c2CCC3)=O)C1C c1(C(N2CCC(C3N(C(c4c(C)nc[nH]4)=O)CCC3)C2)=O)ccc2ncsc2c1 C1(NC(C=CC(CC)C)=O)CCN(C(=O)COC2CCC2)CC1CO C1(NC(CN(C)C(C2(F)CCOCC2)=O)=O)CCCC2(CCC2)C1 C1(NC(CC=CC=C)=O)CC2(CCN(C(C3CCCC3c3nncn3C)=O)C2)C1 C(=O)(CCC(C)(C)C#N)NCC1CCCC(NC(CN(CCOC)C)=O)C1 C1(C2CCCCC2)(NC(CN(C)C(C2CCCC(CF)C2)=O)=O)CC1 Cc1cc(C(N2CCC3CCC23CNC(c2cc(Cl)ccc2F)=O)=O)ncc1N CC1CN(C(c2cnc(Cl)c(Cl)c2)=O)CC(C)N(C(=O)CCn2cccc2)C1 C1(CNC(c2c(CC)[nH]nc2Cl)=O)CN(C(c2[nH]cc(C)c2C)=O)CC1(F)F c1(C(=O)NC(C(=O)OC)Cc2c[nH]c3ccccc23)n[nH]c2ccc(O)cc12 c1(-n2c(Cc3cc(OC)c(C)nc3)nc(C3CCC3)n2)ccc2ccccc2n1 C1(NC(c2c(CNC(CC3N(C)CCCC3)=O)occ2)=O)CCNC(=O)CC1 C1(CNC(c2ncc(F)cc2F)=O)CC2(C1)CN(C(=O)COC1CCCC1)C2 c1(C(=O)NCCC2CCCN(C(C(C)SC)=O)C2)[nH]c(C)c(S(N)(=O)=O)c1C CCC(CN(C)C)CC(=O)NC1(CF)CN(C(=O)CCC2CCCCO2)C1 c1(C(N2CC3CCC2CN3C(=O)C(F)(F)CC2CC2)=O)cnn2c1OCC(F)C2 c1(C(N2CC3(C(NC(c4ccc(CC)s4)=O)CC3)C2)=O)cc2c(nn1)CCCC2 C1(C(=O)NCCCCCCNC(=O)C=CCN2CCCC2)CCOC(=O)CC1 C(=O)(CC(C)(C(F)F)N(C)C)N1C(CCOC)CN(C(c2ccsc2)=O)CC1 Cc1coc2ccc(C(=O)NC(C)CC(C)NC(=O)C3=CCOC3)cc12 C(=O)(C(C#N)(CC)CC)N(C)CC1OCCN(C(CN(C2CC2)CC)=O)C1 C1(NC(C2CCN(C(CCC3CC(OC)C3)=O)CC2)=O)CN(C)CC1(F)F Cc1cccc(C(=O)N(C(C)C(=O)N(CC(O)C2CCC2)C)C)c1O C1(CNC(c2nc(C)sc2C)=O)CN(C(c2scnc2C(C)C)=O)C2(CCC2)C1 c1(C(C)(C)C)ccnc(C(=O)NC2CC2CNC(c2cncc(CO)c2)=O)c1 N1(C(C2C3CN(C(c4c(OC)nn(C)c4)=O)CC32)=O)C2CCC1CN(C)C2 c1(NC(=O)NC2CC23CCSCC3)cccc2c1CCOC2 c1(CC(=O)NC2CCCC(CNC(CCCC=C)=O)C2)ccc(Cl)c(F)c1 C1(NC(=O)C=CC(F)(F)F)C=CCN(C(c2ccn(C3CCC3)n2)=O)C1 C1(C(N(CCN(C(c2[nH]cc(C)c2)=O)C)C)=O)CCC(C(C)(C)O)CC1 N1(C(c2cn(C3COCC3F)nn2)=O)CC(O)(C2(CNC(C3CCO3)=O)CC2)C1 Cc1nc(C(=O)N(C2(CO)CCCCC2)C)cn1C.C1(C)C(=O)N1.CCF c1(CC)oncc1C(=O)NC(C)(CNC(c1nncs1)=O)C1CC1 CC(C(=O)NC1CCC1NC(=O)C=Cc1ccc(C2OCCO2)o1)C(F)F C(=O)(C(C)CCCC(C)=O)NC(C(=O)NC(CNC(=O)OC)C)CCC(C)C c1(C(=O)NC)c(C)o[nH]c1=NC(=O)Oc1cccc(C(N2CCOCC2)=O)c1 c1(OC)ccccc1NC(C)C(CO)NC(c1ncccc1NC1CCC1)=O C1(NC(c2c(C)oc(Cl)n2)=O)CCN(C(c2ccc(NCCO)cc2)=O)CC1C c1(CN2CCC(C3(NC(CCCC)=O)CC3)CC2)ccnc2ncnn12 Cc1ccc(C=CC(N2CCN(C(=O)C(CO)c3ccccc3)CC2)=O)cc1C c1(C(N(C2CN(C(Cc3c(C)ccs3)=O)CC2F)C)=O)ccc2c(c1)CCO2 C1(c2ccccc2)(COC(C(C)SC)=O)CCCO1.C1(=O)CO1 C12(NC(C3(C#C)CC3)=O)CCCN(c3cc(CC(C)C)ncn3)CC1C2 C(=O)(C1=CSCCO1)N(CCCNC(CC1CCCC(C)C1)=O)C1CC1 CCCC(CCNC(C1(C2CC2)CCCO1)=O)CNC(=O)COCC(F)F C(C)(CO)(C(=O)N1CCC(CO)(CNC(=O)COC(C)(C)C)C1)OC Cc1ccc(C(F)CNC(=O)NC(C2(F)CC2)C)cc1F c1(CC(=O)NC2CC(C(=O)NCCCS(C)(=O)=O)C2)cc([N+](=O)[O-])ccc1F C(=O)(C1CCSc2ccccc21)NCC1(NC(C2=NOC(C)(C)C2)=O)CC1 c1(CC)cc(C(N2CCOCC2C2CCC2)=O)ccc1OC(F)(F)F n1(CCC)cc(C(=O)NC2CC(CCC(N3CCOC3C(C)C)=O)C2)nn1 CC1(C)CC(NC(C2CC=CCN2C(=O)C(=O)NC2CC2)=O)CO1 c1(-c2cn(CC(C3OCCC3C)C)nn2)ccc(COOC(F)(F)F)cc1 Cc1cc(N2CCCNC(=O)C2)nc(N(C)CC2CCOC2C)n1 C1(S(C)(=O)=O)(C(N2CCN(C(c3c(CC)n(C)nn3)=O)CC2)=O)CC(O)C1 CCCCCCC(C)C(=O)NC(C)C(CO)NC(c1cccc(CCO)c1)=O C(=O)(C(CC1CC1)NC(=O)NCCC1(C)CC1(F)F)OC n1(CC(=O)NCC2(CNC(C(CCCC)C)=O)CC2)nnc2c1CCCC2 c1(NC(C2(CCC=C)CN(C(c3c[nH]nc3C)=O)C2)=O)cc(C)ccc1C C1(C(=O)NCC2(C(=O)NC3C=CCCCC3)CC2)CN2CCN1CC2 c1(CNc2cn(C)c(C(=O)N=c3cc[nH]cc3Cl)c2)ccc(O)c2ccccc12 C1(CNC(C2CC(NC(CCC)=O)C2)=O)CCN(S(=O)(=O)C(F)F)CC1 n1(CC(=O)NC(CNC(c2ccc(C#C)o2)=O)C)nc(C(F)(F)F)c2c1CCC2 C(=O)(C(CN(C)C)CC)N(C(Cn1cc(C(C=C)(C)O)nn1)C)C c1(C(N2CC(NC(c3csc(=N)[nH]3)=O)CC(C)C2)=O)ccnc2cc(F)cnc12 C1(NC(CCCC)=O)C2CC1N(C(c1cc(C3(C)COC3)no1)=O)C2 C1(C(=O)NCC2CN(C(c3cccc(C)c3C)=O)CC2C)CN(C)C(=O)CCO1 C(=O)(C(F)(F)CC(C)C)NCC1N(C)CCN(C(C(COC)OC)=O)C1 C1(c2n(CCCSCC)nnn2)(NCc2c(C)coc2C)CC(C)CC(C)(C)C1 C1(NC(=O)CCc2cnc3ncccn23)CCc2nnnn2CC1 C1(C(N2C(CC(=O)NC3(C=C)CCOCC3)CCC2)=O)CC(=O)CC12CCC2 C1(CNC(c2cnn3cccnc23)=O)CC2(CCC2)CN1C(C1CCC=CO1)=O N1(C(CNS(CC)(=O)=O)=O)CCC(O)(CCNC(C2C=CCC2)=O)CC1 c1(CC)nccn1CCNC(=O)C(c1cccs1)NC(=O)CCCF c1(CCC)cc(C(=O)NCCN(C(c2ccc(C3CC3)cn2)=O)C2CC2)c(C)o1 C12(CNC(C(C)OCCC=C)=O)CCC1CN(C(=O)CCc1ccncn1)C2 CC1CC(C)N(C(c2cnc3sccn23)=O)CCN1C(=O)CC1OCCO1 CC(CCCCNC(=O)CCC1CCCN1C)NC(C1CC1(F)F)=O C(C(C)C(=O)NCC#CC(=O)NCC(C)N(C)C)OC(C)=O c1(COC(CCC(N)=O)=O)ccc(Br)cc1F N1(C(CC(CNC(c2c(CC)nccn2)=O)O)=O)CC2CCC(O)CC2C1 c1(C(N(CC(N2CCC(O)C2)=O)CCC)=O)ccc(C2CC2)cc1.N(C)(C)C C(CC(C)CCNC(c1cnn(CC2CCCCC2)c1)=O)NC(C=CC(C)C)=O c1(OC)cccc(F)c1C(=O)NCCOCCn1cnc(Br)c1 c1(C(N(CCNC(CCOCC(C)C)=O)C2CC2)=O)cc(Br)sn1 c1(C(N2CCCC(O)C2)C(=O)Nc2ccccc2C)c2c(nn1C)CCOC2.CS c1(C(=O)NC(CNC(CCCCC(=O)NC)=O)CO)oc2ccc(Cl)cc2c1C C1(NC(c2cnco2)=O)CN(C(=O)CCCc2cnccn2)CC1CO c1(CC(=O)NCC(C)N(C)C(C2CC=CC2)=O)cocn1 CC(C)CC(CNC(C1CNC(=O)N1C)=O)NC(=O)COCCC1CCCC1 C1(C2CCN(C(c3cc(C)c(C)o3)=O)C2)(NC(C(C(CC)C)O)=O)CC1 c1(CCC(=O)NC(CC=C)CNC(=O)C(C)(C)C2CC2)cccc(F)c1 C1(CNC(C2OCCN(C)C2)=O)CC2CCC1N(C(C13CCCCC1C3)=O)C2 N1(C(Cc2c(C)cco2)=O)C2CCC(C2)C1CNC(=O)CC1CCOCC1 c1(C(N(C(C(=O)O)C2CCOC2)C)=O)cnc2c(c1)c(C(F)(F)F)nn2C N1(C(C2(CS(N)(=O)=O)COC2)=O)CCCC(C2CCCN(C(C3(F)CC3)=O)C2)C1 c1(CC(=O)NCCOCCC(=O)NC2(CC(C)C)CCC2)cn(C)cn1 C12(CNC(C(C=C)O)=O)CC(CC)(CN1C(=O)CNC(c1cncc(Cl)c1)=O)C2 C1(CC(N)=O)(NC(C(C)NC(N)=O)=O)CCN(C(=O)CC2CC(C)(C)CO2)CC1 C=CCCC(N)C(=O)NC(c1ccccc1O)C c1(OCC)ccc(C(=O)NCC(C)(C)CNC(=O)CCCC(F)F)c(F)c1F Cc1cc(=O)oc(C)c1C(=O)NCCc1cn(-c2ccc3sccc3c2)nn1 C1(C(=O)N(C2CC(F)(F)C2)C)(CNC(c2c(C)noc2)=O)CC12CCC2 C1(CC=C)(NC(C2CCC(=C)CC2)=O)CCN(C(=O)C=C(Cl)Cl)C1 c1(C(=O)NCCC(C)NC(C2(C(F)(F)F)CCOCC2)=O)occ2c1CCCC2 S(=O)(=O)(c1cnc(NC2CCCc3ccoc32)c(Cl)c1)NC1CCCS(=O)(=O)C1 C1(C(NOCC=C)=O)CC2CCC(C1)N2C(C1OC2CCC1C2)=O C(=O)(C(F)(CNC(C12C(=O)C3CC1C2C3)=O)C(C)C)N1CC(C(=O)NC)C1 N1(C(CCc2ccc(C)s2)=O)CCCCC1C1(NC(C23CCC(C2)C3)=O)CC1 C12CC(F)CN(C1)C(=O)C(C(C)C)N2.c1(OC(C)C)cccc(C#N)c1 C1(n2ccnc2)(C(=O)NCC(CNC(C(c2cnn(C)c2)OC)=O)C)CCCC1 C1(CC=C)(NC(C2CC=CCO2)=O)CCCN(C(c2cnc(Br)s2)=O)C1 C1(NC(CSC)=O)(CNC(c2cccc(C)c2O)=O)CC2CCC1C2 CC(C)(C)CCCCC(=O)N1CC2C=CC1C(C(N1CC(c3ccon3)C1)=O)C2 C1(C(=O)NCC=O)(CO)CC(NCC2CCCC2)C1.C1(C2CC2)CC1.C(=O)(N)N N1(C(c2nc(OC)c(C)s2)=O)CCCC(C2(NC(=O)C(C)N(C)C)CC2)C1 c1(SCC(=O)NCCNC(C23CCCC2(CO)C3)=O)cccc2cccc(Cl)c12 CN1CC(C)(C)CC1C(=O)NCCC1(NC(=O)C2=COCCC2)CCC1 C#CCCCCCC(=O)NCC1CCC(C)N(C(=O)CC2CCC(C)(C)O2)C1 Cc1ccc(C(=O)NC(C)CNC(=O)C(C#N)C2CC2)cn1 c1(C(=O)OCC)coc(C=CCN(C)CCC2CCCCO2)c1 C(=O)(C(C(C)C)n1cccc1)N(CCn1cc(CC(C(C)C)O)nn1)C1CC1 N(C1CCc2ccc(F)cc21)C(CC(C)C)c1n(CCCCCC)nnn1 C1(CNC(C(CNC(C(C(C)C)C2CCC2)=O)N(C)C)=O)CC12CCCCC2 N1(C(C(OC)OC)=O)CCOC(C2CN(C(C3(CO)CC3(C)C)=O)C2)C1 c1(C(=O)OC)cccc(C(N2CC(CC(C)NC(=O)C=Cc3cn[nH]c3)C2)=O)c1 c1(C(C(=O)NCCCSC)(C)N(C)CCOCCN(C)C)ccc(Cl)cc1F c1(C(=O)NCCOCCOCCNC(C2CC2C2CC2)=O)cc(F)ccc1Cl C1(C(=O)NC2CC=CCC2)(CC)CCCN1C(=O)CC1(O)CCOCC1 C1(NC(CN(C)C(=O)C2CC2)=O)CC2C(C1)C2(C)C c1(C(c2n(CCCSC)nnn2)NC(C2CCCCC2)C)cn(C)nc1C(F)F C1(CC)CN(C(c2cc(C3CC3)cc(F)c2)=O)CCN1C(=O)C(C)OCOC c1(CC(C(=O)NCCCO)NC(c2ccc(C)o2)=O)ccccc1Br c1(N(Cc2nc(CC(=O)NC(COC)C)sc2)CC2CCC2)cccc(F)c1Cl C1(C(=O)NC2(CN(C(=O)C=Cc3cccc(CO)c3)C)CC2)COCCC1(F)F Cc1nc(SCC(=O)NCC(CO)NC(=O)CCc2ccnn2C)n[nH]1 Cc1nccnc1C(N1CC2C(CNC(C3C=CCC3)=O)C2C1)=O c1(N2CCN(CCNC(C3C(C)CC4CC4C3)=O)CC2)ncccc1[N+](=O)[O-] C12(NC(CCc3c(C)ncs3)=O)CCC(C1)N(C(C1(C)C=CCC1)=O)C2 c1(NCC2(Br)C(F)(F)C2)cc(Cl)nn2cnnc12 CC1CN(C(=O)C2=NOC(C)(C)C2)CC(C)N1C(=O)C(c1ccc(F)cc1)(F)F c1(CCC(N2CC3C(N(C(C(C)SC)=O)C)C3C2)=O)ccc(Cl)c(Cl)c1 N1(C(C2C(C)(C)COC2)=O)CCC=C(CNC(=O)CCC(F)(F)F)C1 C1(COC)(NC(=O)C2=CCOCC2)CCN(C(=O)C(C)NC(=O)NC)CC1 Cc1nn(C)c(C)c1CNC(N1CC(O)(C2CCC(=O)N2)C1)=O Cc1cc(C(=O)N(C(C)CNC(=O)CC2CCC(C)(C)C2)C)c2c(C)n[nH]c2n1 c1(N2CCC(CNC(c3cnc(F)c(F)c3)=O)C23CC3)ncnc2c1CCCC2 N1(C(c2nc(OC)oc2)=O)CCCC(C(C)(O)CNC(=O)C=CCOC)C1 C1(NC(c2ccc(SC3CC3)s2)=O)(CO)CCCN(Cc2nnc(C3CC3)s2)C1 c1(OCCCOC)cc(OC)cc(C(=O)NCC#CCNC(=O)C2=CCCS2)c1 N1(C(=O)CCC2CCCCC2)CCCC(C2CCCN(CCC3CCOC3)C2)C1 Cc1cnnc(O)c1C(=O)NCC1C=CCN1C(c1cccn(C(F)F)c1=O)=O N1(C(=O)OC(C)(C)C)CCC(C2CCCN(Cc3cnc4c(F)cccn34)C2)C1 N1(C(CSCC)=O)CCC2(NC(c3ncc(C)cc3F)=O)CCCCCC12 C1(NC(c2ccc(OC)s2)=O)(CO)CCN(C(c2cc(C3CC3)on2)=O)C1 c1(NC(=O)C(C2CCN(C(=O)C=CC(=O)OCC)CC2)O)ccc([N+](=O)[O-])cc1 C1(NC(C(CC=C)(F)F)=O)CN(C(c2cc(Cl)c(N)cc2F)=O)C2CCCCC12 C=CCC(CC(F)F)C(=O)N1CC(C(C)NC(=O)C(C)SCC)C1 c1(OC)cc(C(N2CCC(C)(C(=O)NC34CCCC3OCC4)C2)=O)cc(C)n1 c1(CNC(c2nc(NC(C(CCC)OCC)=O)sc2)=O)cccc(Br)c1C N1(C(c2cc(OC)cc(C)c2)=O)CCCC2(CCC2NC(=O)CCOC(C)=O)C1 N1(C(c2ncn(CC)n2)=O)CCSCC1C(=O)NC(c1cccc(F)c1)C N1(C(C(C)NC(N)=O)=O)C2CCC(C2)C1CC(=O)NCC(C)(C)CN=[N+]=[N-] c1(C(N2CC3C(NC(C4CC(OC)C4)=O)(CC3)C2)=O)ccc2ccn(C)c2c1 C1(C(N2CCC(N(CCC)C(c3ncccc3F)=O)C2)=O)COCCC1(F)F c1(C(=O)NC(CCNC(CC(C(=C)C)O)=O)C)c(C)nn2cc[nH]c(=O)c12 c1(C(N(CCNC(CN(S(CC)(=O)=O)C)=O)C2CC2)=O)cccc(C(C)(F)F)c1 c1(C(C)NC(c2cccnc2)=O)nocc1C(=O)N(CC(F)F)CCO C1(C)(CNC(N2CCN(c3snc(CC)n3)CC2)=O)CCOC2(CCC2)C1 C1(OC)CC2CC(C(=O)Nc3oc(CNC(C4(CN(C)C)CC4)=O)cc3C)CC12 N1(C(CCOc2cccc(C)c2)=O)CC2CC1CCN2C(C1CCCSC1)=O N1(C(CC2C(C)(C)C2)=O)CCCCC(NC(C2C=CCS2)=O)C1 C1(NC(c2ccc(Cl)cc2)=O)CC2(C1)CN(Cc1cccc(Br)c1F)C2 c1(N(C)CC2CCCO2)nc(N2CCN3CCCC3C2)c2c(n1)CCS2 O=C1CCC(C(=O)N2CC(NC(=O)Cc3nc[nH]n3)C(O)C2)c2ccccc21 c1(C(=O)NC2CN(C(CC=C)=O)CC2C)ccc(C(C)CC)nc1O C(=O)(CCCCC(=O)NCC1CC1NC(=O)C(F)(F)c1cnccn1)NC C(=O)(N1OC2C=CC1CC2)C1C(NC(=O)CCC2CCCO2)CC1 C12(CNC(Cn3c(=O)ccc(C)c3)=O)CCCC1N(C(=O)CC1CCC1)CCC2 C#Cc1ccccc1CC(N1CCCC1CNC(=O)C(F)F)=O c1(CC(N2CCC(O)(C(C)NC(c3ccc(Cl)cn3)=O)C2)=O)cccc(N)c1N C1(C(N2CC(CNC(C(C(C)C)N(C)C)=O)OCC2)=O)CC12CCCCC2 Cc1cc(F)c(CC(N2CC(F)CC2CNC(=O)C(C)C(F)F)=O)cc1F N1(C(c2cn(CC)nn2)=O)CCOCC1CCNC(=O)C(C)c1cncs1 CCC(C)(COC)CNC(=O)CC1(N(C)C(C2(C)CC(C)C2)=O)CC1 N1(C(C2(N=[N+]=[N-])CC2)=O)CCN(C(c2sccc2Cl)=O)C2CC12 C1(O)(CC)CCCN(C(c2sncc2Br)C(=O)NC2CCCC2)C1 c1(C(=O)NCC(CC)NC(c2ccnn2CCN(C)C)=O)cncc(OC)n1 c1(C(=O)NC(C)C(C)NC(c2coc(CO)c2)=O)cc(S(N)(=O)=O)c[nH]1 c1(CC)cc(CN2CCC(CC(N3CCOC4CC34)=O)C2)ccc1C N1(C(CN(C)S(N)(=O)=O)=O)CCC2OCCN(C(=O)C(C3CCCCC3)F)C2C1 C(=O)(C(F)C(C)C(F)(F)F)N(CCN(C(C1CCC(=C)CC1)=O)C)C Cc1cc2c(C(=O)N(CCC(C)NC(=O)C(C)CC3CC3)C)nccn2n1 N1(C(c2cc(CC)nn2C)=O)CC(C)(C)OCC1CNC(C1CCCCC1O)=O c1(C(=O)NCCN(C(C2(S(C)(=O)=O)CC2)=O)CC)ccc(Cl)c(OC)c1 C1(C#N)(CC)CCN(C(=O)C=CC(C)(C)N(C(=O)CC2CCCO2)C2CC2)CC1 C(=O)(CCCCCCC)N1CC2C(N(C(CC(C=C)OC)=O)C)C2C1 CC1CC(NC(=O)C(F)(F)F)CN(Cc2ccccc2CCC(=O)O)C1 c1(C(=O)NC(CNC(Cc2c(SC)cccc2)=O)C)cc2ccncc2c(O)n1 C1(N(C(C2(C(F)F)CC(=C)C2)=O)C2CC2)CCCN(C(=O)C(=Cc2ccco2)C)C1 c1(SCC(=O)N(C(CCNC(C2C(C)(COC)C2)=O)C)C)ccncc1 N1(C(C(n2cc(C3OCCO3)nn2)C)=O)CCOCC1c1cnccc1C(=O)O c1(C(=O)NC2C(C=C(C)C)C2(C)C)ccc(Oc2ccc(Cl)nn2)cc1C N1(C(CC=CC)=O)CCn2ncc(S(C)(=O)=NC(=O)C3(CO)COC3)c2C1 Cc1cc(=NC2CCN(C(=O)CC3CSC3)C2)[nH]c(-c2ccccn2)n1 c1(NC(C)=O)cc(C(=O)NC2CN(C(=O)CC3CC3(Cl)Cl)CC2(C)C)ccc1F C1(CC=C)(NC(c2ncn(C(C)(C)C)n2)=O)CN(C(=O)C(C)N(C)C)C1 N1(C(Cc2cnc(C)s2)=O)CCC2C(NC(=O)CCN3CCC(C)CC3)C12 c1(C(=O)NC(c2cn(Cc3c(C)c[nH]n3)nn2)CC(N)=O)cccn(C)c1=O C1(C)(CC(=O)NC2(COC)CC2)CCN(C(c2c[nH]cc2C(C)C)=O)C1 CC1C(O)CCCN1C(C12C(NC(c3cnn(C)c(=O)c3)=O)C3CC1C2C3)=O c1(C(N2C(C(=O)Nc3c(Br)ccc(C)n3)CC(O)C2)=O)ccc([N+](=O)[O-])cc1Br CCCCCC(O)C(=O)NC(CNC(=O)CCN(C)C(C)=O)CO C1(NC(C(CC2CC2)NC(c2c(NC)scn2)=O)=O)CCCC2(C1)N=N2 n1(CC(=O)NCC(C)NC(C2(O)CCC(C)(C)CC2)=O)nc2ccccn2c1=O CCCC(CC(=O)NC1CN(C)CC1(C)C)NC(=O)COCC(C)(C)C c1(OC)ccc2c(c1)CC(C)N(C(C1Cc3ccccc3C1)=O)C2C c1(CN2C(C(=O)NC(CC)C(F)(F)F)CC3CC32)cccc(Cl)c1F N1(C(COCC)=O)CCCC(C2CCCN2C(=O)CCOC)C1 c1(C(N(CC(C)N(C(CCOC(C)C)=O)C)C)=O)cnoc1C1CC1 c1(CCC(=O)N(CC(C)NC(=O)CC2CC=CC2)CC)cccc([N+](=O)[O-])c1 C(=O)(CC(C)P(C)(C)=O)NCC(C1CCC1)NC(c1c(C)oc(C(F)(F)F)n1)=O Nc1cc(F)cnc1C(=O)NCC1CCN(C(c2[nH]nnc2C2CC2)=O)CC1 N1(C(C(C=C)OC)=O)CCCN(CCNC(=O)C(C)OC)CC1 C1(F)(C(=O)NC(C=CC(=O)NCCCN(CC(C)C)C)C)CCOCC1 C1(NC(CN(CCC#C)C)=O)CCCCN(C(c2cccc(C(C)C)n2)=O)CC1 N1(C(C(CC)C)=O)CC2COCCC2(NC(c2cccc(NS(N)(=O)=O)n2)=O)C1 N1(C(c2cnc(O)cc2O)=O)CCC2C1CCCN2C(c1ccc(Cl)cc1Br)=O N1(C(=O)C(O)C2CCC2)CCN(CCCNC(=O)C(F)(F)c2nccs2)CC1 CCC(O)CC(=O)N1CC(CNC(C2(O)CCOCC2)=O)C1 N1(C(c2ccc(CSCCOC)o2)=O)CCN(NC(C2CCCN2N=O)=O)CC1 N1(C(C(CCC)C)=O)CC(NC(c2ccc(C)c(C)c2)=O)CC12CCC2 C(=O)(CCCCC#N)NCC(N(C(c1cc(OC)ncc1)=O)C)C1CC1 C1(C(=O)NCCCC2(NC(c3[nH]c(=NCC)sc3)=O)CC2)CC12CCCCCC2 C#CC1(CNC(=O)C(O)CNC(=O)C(C)(O)CCN(C)C)CCOCC1 c1(C(N(CC(C)NC(=O)CC2CCC(F)(F)CO2)C)=O)nccc2ncncc12 CC1=C(C(=O)NCCN(C(C2C(c3n[nH]c(C)n3)C2(C)C)=O)C2CC2)CCCC1 N1(C(=O)CC2C=CCC2)CCC2(CCN(Cc3ccc4c(c3)COCC4)C2)C1 CC1C(NC(c2ccon2)=O)CCN1C(=O)CN(C)Cc1cccc(Cl)c1 C1(C(=O)NCCCn2cc(C(=O)NC(c3ccccc3)C)nn2)CCCS1(=O)=O c1(C(=O)NC2CN(C(C(CCC)CCC)=O)C2)cncc2c(OC)cccc12 C1(CNC(c2[nH]c(=NC3C(C)C3)sc2)=O)COc2ccccc2O1 Cc1ccc(NC(C2C3CN(C(c4ccc(O)c(Cl)c4)=O)CC23)=O)c(C)c1Br c1(C(=O)Nc2nn(CC)c(C)c2)cc(-c2ccccc2)nc2ccc(C)cc12 C12(NC(C=C(C)C)=O)CCCC1N(C(=O)C(N=[N+]=[N-])C(C)C)CCC2 CN1CCCC(C(=O)NCc2ccc(C(=O)NCC#CCCO)cc2)C1 N1(C(C2N(CCC#C)CCC2)=O)CC2CC(CNC(=O)CCCCC)CC1C2 N1(C(c2c(C)csn2)=O)CC2CCC(CNC(=O)C(C)(C)C3CCOC3)C2C1 C(=O)(CC1=CCN(C)CC1)N(C1CCN(C(C(C)NC(c2cccs2)=O)=O)C1)C CN1CCCC1(C)C(=O)NCC(C1CCCCC1)NC(=O)CC1CCSCC1 CCCCC(C(=O)NC1(C)CN(C(=O)C=Cc2ccoc2)C1)C(C)C C(CC(O)CNC(c1cn(-c2ccccc2)cn1)=O)NC(c1ccon1)=O CCCCC(CC)CCC(=O)NC(Cc1cccc(F)c1)CC(=O)O C1(C(CC)(C)C)CCC(CNC(=O)CCc2ccc(CC(=O)OCC)cc2)CC1 C1(C(=O)OC)CS(=O)(=O)CN1C(c1cc(CC(=O)OC(C)C)cs1)=O N1(c2c(C)c(Cl)ccn2)CCc2cc(F)cc(Cl)c2C1 C(=O)(CCCCC(N)=O)NCCCC(C)NC(C1CCN(S(C)(=O)=O)CC1)=O CCCCCC(O)C(C)C(=O)NCC1CN(C(c2sccc2Cl)=O)CCO1 C1(NC(C(=O)NCC)=O)CCN(C(c2ccc(N(C)C)nc2)=O)CCC1COC CCCC(O)C(=O)NCCCC(C)NC(c1ncccc1C(C)(C)C)=O C1(C(C(=O)NC(c2nocc2C(=O)NCC2(Cl)CC2(F)F)C)F)CCCCC1 C1(NC(COC(C)(C)CNC(=O)CN2CCCCC2)=O)CS(=O)(=O)CC1C(F)(F)F c1(OC)ccc(NC(=O)C=CCC(C)(C)NC(C2CCCC2C)=O)c(C)c1 n1(C)cc(C(=O)OC)nn1.C(=O)(C1C2CN(C2)C(=O)N1)NCC.C(C)(C)C C1(C(=O)NC2CC(C)(NC(c3cnc(C(C)C)n3C)=O)C2)C2CS(=O)(=O)CC12 c1(C(N(CCCCCNC(C2CC(C#N)C2)=O)C(C)C)=O)cc(Cl)c(Br)[nH]1 c1(-n2c(C(C)COc3cc(F)ccc3Cl)nc(CO)n2)ccc2ccccc2c1 N1(C(CCCN(C(C)=O)C)=O)CCCC(O)(CNC(=O)C(F)(F)C(F)F)CC1 CC1CN2CCN1CC2C(=O)NCC1CCN(c2ccnc(C3CCCC3)n2)C1 N1(C(C2C(C)(C)OC(=O)N2)=O)C2CC=C(C(=O)NCCCN3CC=CC3)C1CC2 C(=O)(C(O)C(C)(C)C)NCCCN(C(=O)CC1(O)CCOCC1)C CCC(C(=O)NCC1CC(NC(C2CC23CCCC3)=O)C1)C(C)C CCC(C)(C)CC(=O)NCCCCCn1cc(C2(F)CCC(COC)CC2)nn1 C=CC1(C(N2CCC(CC(C)C)C2)=O)CCN(C(=O)CC(C)(C)O)C1 C1(C(N2CCC(N(C(=O)CC34CCCC3C4)CCC)C2)=O)CC2C(C1)C2(C)C c1(C(N2C(CCNC(c3cn(CCCF)nn3)=O)CCC2)=O)ccc(Cl)c(O)c1 C#CCCC(C(=O)N1CCC(NC(=O)CC)C1)NC(c1oc(CC)nc1C)=O c1(C(=O)NCC2N(C(c3cnc(C4(C)OCCO4)s3)=O)CCC2)nc2ccccc2[nH]1 CCC(CC)C(F)C(=O)N1CCCC1C(C)(C)C(=O)NCCC(C)OC C1(CCNC(C(C)(C)C)=O)CN(C(C2Cc3ccccc3S2)=O)CCS1(=O)=O c1(CNC(C2CCC2COC(C2(N(C)CC)CC2)=O)=O)ccc(N)c(C)c1 C1(C(N2C(COC)CC2)=O)CCCCN1C(c1ccc(C)o1)=O Cc1cnc(CNC(c2cc(-c3cccnc3)nn2C)C)c(Br)c1 C(C)(CN=c1[nH]ccn2nnnc12)NC(COC1C(C)CCCC1)=O C1(c2nnnn2C2CCC2)(NCc2ccc(OC)c(F)c2)CC(C)NC(C)C1 c1(C(N(CCC)CCNC(=O)CC(O)c2ccccc2)=O)c(Cl)cnn1C(C)C c1(C(=O)NC2CN(C(c3cnn(C(C)C)n3)=O)C(C)CC2)cc(O)c(F)cc1N C#CCC(CC(=O)NC(C1CCCOC1)(C)C)NC(=O)C(C)(Cl)Cl C1(NC(c2c(COC)cc[nH]2)=O)CN(C(c2cccc(F)c2)=O)CC1S(C)(=O)=O N1(C(C(C)OC)=O)CCC(CNC(=O)CCCC2CCCCO2)(OC)CC1 C1(CC=C)(NC(c2oc(CC)nc2C)=O)CCN(C(=O)COCC)C1 c1(OC)cc(NC(C2CC23CN(Cc2cc[nH]n2)C3)=O)c(F)cn1 N1(C(C(C)(C)S(C)(=O)=O)=O)CCC2(CCC2)C(CNC(=O)C2=CCCCO2)C1 Cc1cc(CC2(C(=O)N(C)CCNC(C3(F)CC=CC3)=O)CC2)ccc1F C1(F)(NC(C(C)(C)SC)=O)CCN(C(=O)COc2ccc(C(C)C)cc2)C1 N1(C(CCCN(C(C)=O)C)=O)CCC(NC(=O)CC2CCC=CCC2)C(CO)C1 c1(C(=O)NC(C(=O)NCC2CCC(OC)CC2)CC(C)C)cc2ncccc2[nH]1 c1(C(N2C3CN(C(C4(F)C(C)(C)C4(C)C)=O)C(C3)C2)=O)ccc(O)cc1[N+](=O)[O-] c1(C(=O)NCCNC(c2cc(C3(C(F)F)CC3)[nH]n2)=O)ccc(C2CC2C)o1 Cc1cccc(C(N2CCCC2CCNC(=O)CC2CC(C)(C)CO2)=O)c1 N1(C(C2N(c3nc(C)c(F)cn3)CCC2O)=O)CCCC(C)(O)CC1 C1(NC(C(C)(C)c2cccnc2)=O)CCC(Nc2ncc(F)cn2)CC1 CC1CN(C(=O)CC2CC3(CCO2)CC3)CCN(C(C2CCCC2O)=O)C1 C=C=CCCC(=O)NC(CNC(=O)C(n1ccc(Br)n1)C)C1CCC1 Cn1c(C(=O)NC2CC(O)(CNC(C3CSCCS3)=O)C2)cc2ccccc12 CC1(C(=O)Nc2cnccc2CO)CCCN(C(c2ccc(C(N)=O)cc2)=O)C1 N1(C(=O)Cn2cc(Cl)cn2)CC2(CCN(Cc3ccc(F)cn3)C2)C1 C12(CC)COC(COC(c3cccc(-c4cccnc4)c3)=O)(C1)C2 C1(NC(COCC)=O)(COC)CN(C(=O)Cc2cc(C)[nH]n2)C1 N1(C(C2(C)N(C(C3C(C(C)=O)COC3)=O)CCC2)=O)CC(C)OCC1C N1(C(=O)CCc2cnc[nH]2)CCCC(O)(CNC(C23COCC2C3)=O)CC1 c1(-c2cc(C(=O)NC(CC(C)NC(COCC=C)=O)C)no2)ccc(Cl)cc1 c1(C(N2CCC(C)(CNC(C3(O)COC3)=O)C2)=O)cc2ccc(Cl)cc2[nH]1 C1(CC(=O)N(CCCNC(=O)C=CC2CCOC2)C)CC2(CCOCC2)CO1 C#Cc1ccccc1CC(=O)N(C1CCCCN(C(=O)C(C2CC2)OCC)C1)C c1(NC(CC)CNC(C2(C(F)F)CCOCC2)=O)ncnc2c1CCCC2 C1(C(N2CC(O)(CCNC(=O)CC34CCCC3C4)C2)=O)Cc2cscc2C1 C1(C(=O)NC(C(=O)NC(c2cncs2)C)Cc2cn[nH]c2)CCC(C)(C)CC1 c1(CC)ccc(C(=O)NCC2CC(NC(c3ccc(CO)o3)=O)C2)c(F)c1 n1(CC(=O)NCC2C(C(=O)OC)C2)ncc(=O)c2ccccc12 C1(NC(COCCSC)=O)CCC12CCN(C(c1ccc(C(N)=O)cn1)=O)CC2 CC1CCC(C)N1CC(=O)NCC1CC(NC(=O)C(C)OCC2CCCO2)C1 C12(c3n(CC(=C)C)c(N4CC(=O)NC(=O)C4C)nn3)CC3CC(CC(C3)O1)C2 C(CC1=CCN(C(c2[nH]nc3ncccc23)=O)CC1)NC(C1CC12CC2)=O c1(OC)ccc(OCc2ccn(C(F)F)n2)c(C2CC2C(=O)OC(C)(C)C)c1 c1(-c2c(C)ccs2)ccc(C(=O)NCc2cnccn2)c(C)n1 C1(CC=C)(NC(=O)C=C2CCC(C)CC2)CCCN(C(c2csc(CO)n2)=O)C1 c1(OCC)ccc(Cl)nc1C(=O)NCC1CCC(NC(=O)C(O)c2ccsc2)C1 C1(C(N(CC(N)=O)CC)=O)N(C(=O)C(C)n2cccn2)CCC1(C)C Cc1ccc(C)c(C(=O)NC(C2CN(C(=O)C(=O)N(C)C)C2)C)c1 C1(C)(C(CC)NC(=O)NCCc2csc(C3CC3)n2)CCCOC1 c1(OCC)c(CNC(c2nnnn2C(C)C)c2ccco2)cccc1Cl Cc1cc(N)cc(C(N2CCN(C(c3cccs3)=O)CC(CO)C2)=O)c1F C1(C(=O)NC(CC#C)CO)COCCN1C(C1CS(=O)(=O)C1)=O N1(C(C2(C(C)NC(c3ccc(Cl)s3)=O)CC2)=O)CCC(C)(C)C(NC(=O)C2CC2)C1 C1(C(N(C)Cc2cncn2C)=O)C2CC2CN1C(=O)C(CO)N(C)C C(=O)(CN=C(NCC(c1ccccc1)CO)NC1CC1c1ccsc1)NC(C)C N1(C(C2(C(C)=O)CC2)=O)CCC(NC(=O)Cc2cn3c(n2)CCCC3)C(C)(C)C1 C1(CNC(c2c(C)nc(CC)o2)=O)COCCN(C(c2ccc(C(N)=O)o2)=O)C1 c1(C(C(=O)NCC2CC2)N(CCC)C2CC2)cc2c(s1)CCOC2 c1(C(N2CCN(C(=O)C3=CCSC3)CC2c2cn[nH]c2)=O)ccc2nc[nH]c2n1 C1(NC(C2C(C)(C(F)F)C2)=O)C=CCN(C(C2CCCC(=O)N2)=O)C1 C1(CNC(CCC(=O)NC)=O)N(C(C2CCCN(C)C2)=O)CCC1(C)C c1(C(=O)NCC2C(NC(CC3(C)CC3(F)Cl)=O)CCC2)ncc2ccccn12 C1(NC(C(CCC)NC(=O)CC2CC2(C)C)=O)CCn2ccnc2C1 c1(SC)ccc(C)c(N(C)Cc2cn(-c3ccc(Br)nc3)nn2)c1 N1(CC)CC(C(=O)NC2(CO)CCCN(C(C3(CC4CC4)CC3)=O)C2)CCC1=O C(CC(CC)C(=O)NCC1(F)CN(C(c2ccc(=N)[nH]c2)=O)C1)=CC N1(C(c2c(C)coc2C)=O)CCC(NC(=O)COC(C)(C)C)C(CO)C1 c1(OCC(N2CCC(CNC(CC=C)=O)C(C)(C)C2)=O)ccc(S(N)(=O)=O)cc1 N1(C(c2c(CC)n[nH]c2)=O)CC2(C=C(C(=O)N3CCC4(C=CCO4)CC3)CO2)C1 C(=O)(CCCC(=O)NC1(CO)CCN(C(=O)CCCOC(C)C)C1)NCCC Cc1nnnn1CC(=O)NCC(C1CCOC1)NC(=O)CCCOCCOC.CCCO n1(CC)nc(C(=O)NC(C2CCN(C(=O)C(c3cccs3)SC)C2)(C)C)c(C)n1 C(=O)(C(CN=[N+]=[N-])NC(=O)CN=[N+]=[N-])NCC(c1nncn1C)C N1(C(C2CC(OC)OC2OCC)C(=O)NCCC)CCC2(CCCCO2)C1 C1(C(=O)NC2CC(C)(C)N(C(c3cc(N)cnc3Cl)=O)C2)CC2(C1)CC1(CC1)C2 N1(C(c2cc(C)n(C(F)F)n2)=O)CC2CN(C(c3cscc3C(F)F)=O)CCC12 C1(O)(CCNC(C2CC2(F)F)=O)CCN(C(c2ccncc2O)=O)CC1 c1(CN2C(C(N(CC(C)NC(=O)C(O)CF)C)=O)CC2)ccc(Cl)cc1 c1(N2CC(C)(COC)OCC2)nc(N2CC3CC2C3)c2c(n1)CCCCC2 C(=O)(C(C)NC(=O)CC1(NC(C2CCOC2)=O)CCC1)NCC C1(NC(CCCC)=O)CN(C(=O)CC(C(F)(F)F)OC)C2(CCCCC2)C1 C(=O)(C1CCCc2cncn21)NCCC(N1CCN(C)CC1)C c1(C(N(C(C=C)C)C)=O)ccnc(CNC(=O)CCOCC(F)F)c1 N1(C(C(C=C)(C)O)=O)CC2(C1)C(NC(c1ccn(CC)c(=O)c1)=O)CCS2(=O)=O C(=O)(C(C)C(C)NC(C)=O)NCC(COC)(F)F N1(C(CCSC)=O)CCC(CNC(=O)C(Cc2ccccc2)NC(N)=O)C12CC2 CC1C(NC(=O)COC2CC2)CCCN1C(=O)CC1(C(=O)NCC(F)(F)F)CC1 Cc1cnc(C(N2CCCC(CN(C)C(c3csc(CO)n3)=O)C2)=O)cc1C C1(NC(C(CC#C)NC(=O)C(O)CN(C)C)=O)CN(C)CC1(C)C N1(CCC)CCCCC1C(=O)NCCN(C(C12CCC(C1)C2)=O)C1CC1 N1(C(C(=O)NC(C)C)=O)CC2(CCC2NC(=O)C(C)CN(C)C)C1 c1(C(C)=O)ncc(C(=O)NC2(CCNC(=O)C=Cc3ccco3)CCC2)s1 CC1CC(C)CN(C(c2cncc(CNC(c3cnsn3)=O)c2)=O)C1 N1(C(c2cc3ccc(C)cc3nc2)=O)CCCC(N=c2nc(C)[nH]s2)(CN)C1 c1(C(N(C(CCCN(CC)CC)C)C)=O)ccc(Br)c(Cl)c1 c1(NCC(CCC)(C)C)[nH]c(=NCC23CCCC2OCC3)nc2c1ncn2C C(=O)(C1CCCc2n[nH]cc21)NCC1CCC2CN(C(c3c(C)cco3)=O)CC21 C1(CNC(C2(COC)CC(F)(F)C2)=O)CN(C)CCN1C(c1ccc(C)nn1)=O c1(C(=O)NC(CC(C)NC(c2ncc[nH]c2=O)=O)C)c[nH]c2nc(F)ccc12 CC1(C)CC(NC(=O)CN=S(C)(C)=O)CN1C(C1CC2(CCC2O)C1)=O c1(C(N2CCCC(CN(C)C(=O)OC(C)(C)C)C2)=O)n[nH]c2ccc(Cl)cc12 C1(CC)(OCC(=O)N(CC(C)(C)C)C(C)C)CCC(c2ccccc2)CC1 C(=O)(CC(C(F)F)NC(c1nc(Cl)oc1C)=O)NCCN(OC)C c1(C(N2CCC(OCc3nc(C)oc3)C2)=O)ccc(CN2CCCCC2)cc1 c1(CN2CC3(CC(NC(c4c(OC)cnc(Br)c4)=O)C3)C2)cccc2[nH]ncc12 C(CCC(O)C(=O)NCC(C)F)NC(C(C)SCCCC)=O CC(C)CCC(F)C(=O)N1CCCC(C)C1CCNC(c1cccc(F)c1N)=O c1(OC)cc2cc(COC(C3CCCN(CC(C)O)C3)=O)oc2cc1OC C12(C(N3CC(CC)C(NC(c4cnn[nH]4)=O)CC3)=O)CC3CC(C1)CC(C)(C3)C2 c1(C(=O)NCCC(C)NC(C2CC(C)(C)CO2)=O)cc(Cl)c(Br)[nH]1 CCC(C(=O)NCCN(C(C1(NC(C)=O)CC1)=O)CC)C(F)(F)F C(c1cn(C)c2ccccc12)=CC(=O)NCCC(C)N(C(=O)C(O)C(C)(C)C)C Cn1nc(C(N2CCCC(F)(CNC(C3CCCSS3)=O)C2)=O)ccc1=O C1(COC)(NC(C2CCCN2C)=O)CCN(C(=O)C(C)=CC(C)(C)C)C1 N1(C(C(C)SCCCC)=O)CC(NC(c2cnns2)=O)C(c2cncn2C)C1 c1(C(=O)NCC(C)(CO)NC(c2cn(C)nc2Br)=O)noc2c1CCCC2 N1(C(C(CCC)O)=O)CCN(C(c2occc2Cl)=O)C(CF)C1 Cn1ccc2ccc(C(=O)NC(c3ccncc3)C3CC3)cc12 C(=O)(C1=NOC2(CCC2)C1)N1CCC(F)(CNC(C2CC2C2CC2)=O)CC1 Cc1nnc2cnc(C(=O)NCC3CN(C(C4CNC(=O)N4)=O)CCCO3)cn12 c1(Cc2n(CC(=C)C)c(N3CCC(F)(C#N)C3)nn2)cc(F)cc([N+](=O)[O-])c1 [N-]=[N+]=NC1CCC(C(=O)NCC2(CNC(=O)CCC3CCOC3)CCCC2)CC1 c1(CNC(C(c2ccnn2C)NC(C(CCC)O)=O)=O)cnc(F)c(C)c1 N1(C(C2(OC)CCCC(C)C2)=O)CC(C2CN(C(C3(F)CCCCCC3)=O)C2)C1 N1(c2sc(C#N)c(Cl)n2)CC23CCCCC2(CN(C(C2(CO)CC2)=O)C3)C1 N1(C(C=C(C)c2cccs2)=O)CCC2(CC1)CN(C(C1CN3CCCC1C3)=O)C2 C(=O)(C(C)(C)CCNC(=O)CN1CCC(O)CC1)NC(C=C)CO c1(CC(=O)NC(CC)CNC(c2c(C(=O)OC)cnn2C)=O)ccc(C)c(C)c1 C1(CNC(C2CC3CCC2C3)=O)CC2CCC1N(C(=O)C(F)C1CCOC1)C2 c1(C(N(C2CCN(C(c3nccn3C)=O)C2)C)=O)cc2oc(Br)cc2s1 c1(C(=O)NCC(C)N(C(=O)CN(C)Cc2ccc(Cl)s2)C)ccnc(F)c1N c1(CC)n[nH]c(CC)c1CC(=O)NC1CN(C(=O)CC2(C)CC2)CC1OC c1(C(=O)NCCC2CCN(C(CC(CC)(F)F)=O)C(C)C2)cc(N)c(Cl)c(O)n1 c1(CCC(=O)NCC2CC(C(N(C)CCN3CCOC3=O)=O)C2)cncnc1O N1(C(C2CCCC(C)CC2)=O)CC(NC(C2CC(=O)CO2)=O)CC(C)(C)C1 C12(NC(=O)COCc3ccccc3)CC1CN(C(C1(O)CCSCC1)=O)C2 CC1CCCN1CC(=O)NC1(CNC(=O)COCCCF)CCCC1 C1(CC(=O)NCc2c(C)n(C)nn2)CN(C(=O)Cc2cccc(F)c2)CC12CC2 C(=O)(C(O)C1=CCCCC1)NCC=C(C(N1CC(OC)C2(C1)CC2)=O)C CC1CC(CN(C2CC2)CC2(C3CCCO3)CCC2)CCC1=O c1(SC(C(=O)NCC(CC=C)NC(c2csnn2)=O)C)ccccc1Cl N1(C(c2c(C(C)=O)cn(C)n2)=O)CC2CCC1C(NC(=O)C(C)C#N)C2 C12(NC(C3CCCC(C(=O)OC)C3)=O)CCCN(C(c3cc(C)sn3)=O)CC1C2 C#CC1(C(=O)NC(C)C(O)C(C)C)CN(C(=O)COC(C)=O)C1 C12(C(N3CC4CC(NC(c5cc(C)sn5)=O)C4C3)=O)CCCN(CCC1)C2 N1(C(c2cc(C)ns2)=O)CC2CC(NC(=O)CCC3(C)CC3)CC2C1 N1(C(c2nc(C)c(C)s2)=O)CCC2(C)CN(C(c3cc(Cl)ccc3F)=O)CC12 O=S(=O)(c1ccn(C2CCCCC2)n1)N(C1CC1)Cc1cccc(F)c1 S(=O)(=O)(CCC(=O)NC1CN(C(=O)CC(C)(C)O)C2CC12)NC CCCCC(C(=O)N1CC(CNC(c2c(F)ccc(F)c2Cl)=O)C(C)C1)C(C)C CC(C)(C)C(O)Cc1cn(C2CCN(C(c3nscc3Br)=O)C2)nn1 c1(C2CCN(c3cc(N4CC(C)OCC4)ncc3)C2)cccc([N+](=O)[O-])c1 N1(C(CCc2cnn(C)n2)=O)CC(NC(=O)CN2CC(=O)NC2=O)CC2(CC2)C1 c1(N(C(=O)CC(C)C)C(=O)NCC(CNC2CC2F)OC)ccsc1-n1cnnn1 N1(C(C2N(C(c3scc(OC)c3)=O)CC(O)C2)=O)CCS(=O)CC1C c1(C(N2C(CCNC(C(CC)CC)=O)CCCC2)=O)ccc(OC)c2occc12 C1(C(N(c2nc(C(=O)NC3CCN(C(C)=O)CC3)cs2)CC)=O)CCOC(C)(C)C1 Cc1ccc(C(N2CC3(CO)CC2(C(=O)NCCC2CCCC2)C3)=O)cc1CO Cc1csc(=NCC(=O)N2CC(C)(C)CCC2CNC(c2ccc(CO)o2)=O)[nH]1 C1(NC(c2nc(C)c(C)s2)=O)CCN(C(c2ncncc2F)=O)C(C)C1 C1(NC(=O)CCn2cc[nH]c(=O)c2=O)CCC2CC1CN2C(c1cnc(O)o1)=O N1(C(C(CC)O)=O)CC2CCCC1(CNC(c1cnc(C(C)(F)F)s1)=O)C2 N1(C(Cc2scc(C)c2)=O)CCOC2(CCCN(C(=O)CC(C)P(C)(C)=O)C2)C1 N1(C(c2ccc(CC)s2)=O)C(CNC(C2CCS(=O)(=O)N2)=O)CC2CC12 C1(OC)(CNC(c2cocc2C)=O)CCN(C(=O)CC(C2CC2)C2CC2)C1 CON1CCC(CC(=O)NCC2(O)CCN(C(=O)COC3CC=CC3)C2)CC1 c1(OC)ccc(C(N)=O)cc1NC(=O)OC(C)(C)C.c12cc(no1)C(=O)NC2 N1(C(C=CSC)=O)CC2CCCC2(NC(c2cn(Cc3ccccc3)nn2)=O)C1 CC1CN(C(c2ccc(Cl)cc2N)=O)CCCN1C(C1CCCSC1)=O C#Cc1cc(C(N2CC3CC2C3C(=O)NC(C)COCC)=O)ccc1C N1(C(C)C(=O)Nc2ccc(Cl)cc2Cl)CCC2C(=O)NCC2C1 c1(C(=O)NC(C)CNC(c2nc(CN(C)C)no2)=O)ccccc1-n1ccnn1 C1(N=[N+]=[N-])(C(N2CC(C(C)O)C2)=O)CCN(C(=O)CCOC2CCC2)C1 c1(NC(c2nc(-c3cnn4c3CCCC4)cs2)=O)c[nH]c2ncccc12 c1(OC)ccc(CC(=O)NC2CN(C(=O)Cc3cnn(C(F)F)c3)C2)cc1 C1(C(N(CC(F)Cl)C)=O)CC(O)CCN1C(=O)C(C1CCCCC1)F CC(C)CC(F)(F)C(=O)NCC1CCCN1C(C1CCC(F)C1)=O CC(C)(CC(=O)NCCN1CCNC(=O)C1)NC(=O)COC1CCCCC1 c1(C(=O)NC2(CCNC(CCC(C)OCC)=O)CC2)cccc2c[nH]nc12 c1(C(N(C2CCN(C(C(C)OCC=C)=O)C2)CC)=O)onc(C)c1C C(=O)(C(C)(C)C(F)(F)F)N1CC(CC(=O)N(CC(C)OC)CC)OCC1 C1(CNC(CC(c2scc(C)c2)O)=O)CN(C(c2cc(C(C)C)[nH]n2)=O)CCO1 c1(CSC)ccccc1CC(=O)NCC(O)CCNC(=O)C(C1CCOCC1)F CN1N=CC(CC(=O)NC(c2ccc(F)cc2)CNC(C2(C)CCC2)=O)C1=O C1(CNC(=O)Nc2ccc(CS(=O)(=O)N(C)C)cc2)CCCC2(CCC2)O1 C1(NC(CCCN(C)N=O)=O)CN(C(c2cc(CCO)on2)=O)CC2(CCC2)C1 CC(C)(CCCNC(c1ccccc1SC(F)F)=O)NC(=O)CC1CCC(O)C1 C1(C(=O)NCCC2CC(NC(C(C#C)(C)C)=O)C2)CC12CCS(=O)(=O)CC2 c1(OC)ncnc(C(=O)NC(C2CCCN2C(=O)CC2SC(=N)NC2=O)C)c1F C(C(C)(C)CN=c1[nH]nc2ccc(C(F)(F)F)cn12)OC c1(C(N2C(C(=O)Nc3cccc(SC)c3)CC(O)C2)=O)cccn2cncc12 Cc1c(C(=O)NCC23CC2CN(C(C2CC(C)CCO2)=O)C3)c(C(F)F)nn1C c1(COC)ccnc(C(=O)NCC2(F)CC(NC(c3ccnn3C)=O)C2)c1 C1(C2CCN(C(C3C4CCC(=O)C34)=O)C2)(NC(CCc2cnc(C)s2)=O)CC1 Cc1cn2ccnc(C(N3CC(CNC(=O)CSCCC(C)C)CC3C)=O)c2n1 C1(NC(C(CNC(=O)C(c2ccnn2C)O)OC)=O)CC2CC3C(C2)C13 C1(C(=O)NC2CN(C(Cc3nc(C)sc3)=O)C(C)(C)C2)Cc2nnc(C)n2C1 C1(NC(Cc2scc(C)n2)=O)CCN(C(=O)CC2CCCCN2C)CC1C c1(SC)cc(C(=O)NC2(C)CN(C(=O)C(c3cccc(Cl)c3)C)C2)n(C)n1 c1(OC)nn(C)c(Br)c1C(=O)NC(C)CNC(c1csc(C#N)c1)=O c1(-c2n(CCn3c(C)cc(C)n3)ccn2)cc(Cl)ccc1F C1(O)(C(=O)NCCSCCc2ccccc2)CCCN(C(=O)COCCF)C1 c1(C(N2CC(C)(NC(C3CCCC(OC)C3)=O)C2)=O)ccc(CC2CC2)c(C)c1 S(=O)(=O)(c1c[nH]ccc1=NCC1(C)CC2CC2C1)N(CC(CC)(C)OC)C Cc1nc2c(s1)CN(C(C1(C)CC(O)CN1C(C1CC3(CC(=O)C3)C1)=O)=O)C2 n12nc(c(C)n1)C(=O)NCCC1CC(C1)C(=O)N2.c1(C(CSCC)C)cn[nH]c1 CCC(CC(F)(F)F)C(=O)NCC1CC(C)N(C(c2ccn(C)n2)=O)C1 C=C(C)C1OCCC1C(N1CC2(CC2)CC1C(N1CCCC(O)CC1)=O)=O N1(C(C)=O)CCCC2CCCCC12.c1(C(=O)N2C3CCN(C3)CC2)ccc(C#N)s1 c1(CC)ccsc1CNC(=O)CNc1ccc(C(=O)OC)o1 C#Cc1ccc(C(=O)NC2CC(C)(NC(=O)CCC(=O)OC(C)(C)C)C2)cc1C c1(OCCC(N2C(c3cn(CC(CC)CC)nn3)CCC2)=O)ccc(F)cc1F N1(C(CCN(C)CCO)=O)CC2(C1)CN(C(=O)C(c1ccc(Cl)cc1)CO)C2 C=C=CCCC(=O)N1CCC(C(=O)NCC2(CC3CCC3)CC2)(CF)C1 Cc1ccc2c(c1)CCCN2C(=O)NC1CC1c1ccccc1F C(=O)(CCS(C)(=O)=O)NCC(CC(=O)NC1COC(=O)C1)OC c1(CS(N2CCC(C)(O)C2)(=O)=O)ccc(F)cc1Cl CC(C)C(C(=O)N(C)CCNC(c1ncoc1C1CC1)=O)n1cc(Br)cn1 C(CN=c1cc(NCc2ccncc2Br)nc(C(C)C)[nH]1)(C1CCOCC1)OC c1(C(N2C(C(C)NC(CC(C)C(F)F)=O)CCC2)=O)ccc(C#N)c(F)c1 CCS(=O)(=O)CC(=O)Nc1cnc(Cl)cc1C(=O)Nc1n[nH]c(C(=O)OC)n1 N1(C(c2n(COC)ncc2)=O)CCCC(N(C)C(C2CC(C(F)F)C2)=O)C1 N1(C(C(=O)NCC)=O)CCC(NC(c2sc(C)c(C)c2C)=O)C(C(C)C)C1 C1(CNC(CCC2N(C)CCC2)=O)CCN(C(=O)COC2CCCCC2)CC1 C1(C)(COC)CC(NC(c2cccc(F)c2C2CC2)=O)CN1C(c1ccco1)=O c1(OC)c(F)cc(CN2CC(NC(=O)Cc3nnc(C)o3)C(C#N)C2)cc1F c1(OC)cccc(C(N2CCN(C(c3coc(C)c3)=O)C(C)C2)=O)c1N c1(C(=O)NC(C2CCCCC2)C(=O)N(CCC#C)CCO)cn(CCO)nn1 C#Cc1cccc(C(N2CC3CC2C3NC(c2cscc2SC)=O)=O)c1C C(CCN=c1[nH]c(Cl)nc2c1SCC2)NC(C1CC2(CCOC2)C1)=O Cc1cc(C(=O)NC(C)C(C)NC(=O)C=C2CCC(C)CC2)c(N)cc1F C1(O)(CNC(=O)CCn2ccnn2)CN(C(=O)CNC(N2CCCC2)=O)C1 C1(C(=O)NCC2CCN(C(CC)=O)C23CC3)CN2CCCN1CC2 C1(C(=O)NCC2(O)CN(C(C3(C(N)=O)CCC3)=O)C2)CCc2ccccc2O1 C1(NC(c2nccc(CC)c2)=O)CCCN(C(C23CCC(CC2)OC3)=O)CC1 C#CCCN=C(NCC1CC2CCC2C1)N(C)Cc1ccc(Cl)c(OC)c1 Cn1ccc(C(N2CC(CCO)(NC(c3cnn(CCC(F)(F)F)c3)=O)C2)=O)n1 N1(C2CN(C(=O)NCCc3c(C)nccn3)C2)CC(C)(C)OC1=O c1(OCC=C)ccc(Cl)c(C(=O)NCCC(=C)Cc2ocnc2OC)n1.C(=O)OC C1(NC(C=CCC)=O)CC(F)CN(C(=O)C(C)(C)C2CCOCC2)C1 Cc1ccn(CC(=O)NCC2CCCN(C(=O)C(C)(C)CF)CC2)c(=O)c1 c1(C(N2CCC(NCc3ncc(OC)nc3)C2)=O)cc([N+](=O)[O-])cs1 CC1(C)CC(CO)CN(C(c2cc(Br)co2)C(=O)N(CCN2CCOCC2)CCO)C1 C1(C(N2CCC3(CC(NC(C(C)C)=O)C3)C2)=O)CC(c2cccc(F)c2)=NO1 Cc1oc(C(=O)N(C2CCN(C(=O)Cc3cccnc3Cl)CC2)C)cc1CO N1(C(Cc2cccc(OC)c2)=O)CCN(Cc2cc(C(=O)O)ccc2O)C2CC12 Cc1ccc(C)c(C(N2CC(CNC(c3cccc(F)c3N)=O)CCC2C)=O)n1 N(C(=NCC(=O)OC)N(C)Cc1ccc(C(C)(C)C)cc1)CC(COC)(C)CO c1(C(=O)NC(CNC(C(F)=CCC)=O)C)cc(C(F)(F)F)cs1 c1(NC(C2CC(=C)CN2C(C2CCCO2)=O)=O)cc(Br)cc(C(=O)OC)c1C CCC(C)CCC(O)CC(=O)NCCCNC(=O)CCNC(=O)CO C(C(CC(C)C)C(=O)N(C1(COC)CCC1)C)NC(C(C(=O)OCC)OC)=O CC1(C)CCN(C(C2(c3cccs3)CC2)=O)CC1CNC(=O)C1=NNC(=O)CC1 c1(C(=O)NC2CCN(C(c3cc(C4CC4)cc(F)c3)=O)C2)cccc2scnc12 C1(O)(CNC(C2C3CCCC23)=O)CCN(C(c2cn(-c3ncccn3)cn2)=O)C1 C1(NC(c2nnc(C)s2)=O)CCN(C(=O)CN(C)Cc2cccc(Cl)c2)CC1F c1(C(=O)NCC(C)N(C(=O)CN(C)C2CC2)C)cnc2c(c1)CNC2=O C(CC(=O)N1CC(NC(=O)C(=O)NC2CC2)C(OC)C1)(C(F)(F)F)OC C=CC1(C(=O)NC2CC2CNC(c2ccc(F)cc2)=O)CCOCC1 CCC(C)C(O)C(C)C(=O)NC(C)(CO)C(=O)NC1CCOCC1F c12ccc(cc1F)CNC(=O)C(=O)NC2.c1(CNS(C)(=O)=O)ncccn1.C1CC1 N1(C(Cn2ccc(C)n2)=O)CCc2cc(NC(c3ccc(Br)c(F)c3)=O)ccc2C1 C1(CC(=O)NCC(C(C)(C)C)NC(c2cc(Cl)c[nH]2)=O)CCCC2(CCC2)O1 O=C1NCCc2c(C(N3CCN(C(C4CC45CCC5)=O)C4CCC34)=O)cncc21 C(C1=NOC2CCCC12)NC(C(C1CC=CCC1)NC(CC(CC)(F)F)=O)=O C1(NC(c2cnco2)=O)CN(C(c2cc(Cl)ns2)=O)CC1C(F)(F)F CC(C)(CCN1CCOCC1)NS(=O)(=O)Cc1ccsc1 C1(NC(C2CC2CF)=O)CCCN(C(c2c[nH]ccc2=O)=O)C1 N1(C(CCCCN(C(=O)CCc2ccco2)C)=O)CCC2(CCO2)C1 c1(C(=O)NC(CN(C(=O)CSCCOC)CC)C)sc2cc(C)ccc2c1Cl Cc1cc(C)c(C(N2CC=CC(NC(=O)CC3(CO)CC3)C2)=O)cn1 Cn1cc(C(F)=CC(=O)NCC2COCCN2C(=O)CC2CCSC2)cn1 C(=O)(C#CC1CCOCC1)NC1C2(CCN(C(c3c(N)cc(Br)cn3)=O)CC2)C1 c1(OC)ccccc1CC(=O)NC(C)CCN(C(=O)C(C)(C)C1CCCO1)C c1(C(N2CC(CN(C(=O)C(F)CC3CC3)C)OCC2)=O)cc2ccsc2[nH]1 Cc1ncc(-c2cn(C3CCC(C(=O)NCCCN4CCOCC4)C3)nn2)n1C N1(C(CCC)=O)CCCC(C2CCN(C(=O)CN3CSCC3=O)C2)C1 c1(CC)cccc(N2CC(CNC(=O)C(=O)NC(CSC)C3CC3)CC2=O)c1 CN1CCC(CC(N2CCC(O)(CNC(C34COC(C)(C3)C4)=O)C2)=O)C1=O C=CCCCCCCCCNC(=O)C(=O)Nc1cccc(C(N)=O)c1C c1(NC(C2(F)CCN(C(c3ccncc3Br)=O)C2)=O)c(F)c(F)c(Br)c(F)c1F c1(NC(CCC)CCCNC(C2CSCC(=O)N2)=O)ncc([N+](=O)[O-])cc1F CS(=O)(=O)C1CCCN(C(=O)CC(Cc2cccs2)NC(c2ccc(Br)nc2)=O)C1 c1(C(=O)NC2CN(C(=O)Cc3ccsn3)CCC2CO)cc2nn[nH]c2cc1F CON(CCC(=O)N1CC(F)CC1CO)C(=O)c1ccc2nccn2c1 C12(CC(C)NC(C3CCS(=O)(=O)C3)=O)CC3CC(CC(C3)C1)C2 C1(N(C(=O)CCc2ccc(F)nc2)C)CCC(NC(=O)C(C2CC2)N(C)C)CC1 C1(NC(=O)OC(C)(C)C)CN(C(C2CCCN2c2nccs2)=O)CC1(C)C c1(C(N2C(CCNC(C(N3CC(C)C3)C)=O)CCC2)=O)c(Cl)cnn1C(C)C C1(O)CCN(N2CC(NC(c3cc(Cl)c[nH]3)=O)C2)C1.c1(C=O)cc(C(F)F)no1 N1(C(=O)CO)CCC(CCC2CCN(C(C3(n4nccn4)CC3)=O)CC2)CC1 C1(N(C(C(CNC(CC(=O)OC)=O)C)=O)C)CCC(O)CC1 C1(C(=O)NC(CC=C)CNC(C)=O)CCN(c2ccc(Cl)nn2)CC1 CC1CN(C(C2CCCS2)=O)CCN1C(c1cnn(C)c1Br)=O c1(-n2cc(C(C)(C)CNC(=O)CSc3ccccc3Cl)nn2)ccc(F)cc1Cl C1(CNC(c2cn(CC(N)=O)nn2)=O)CN(C(C2C=CC=CC=C2)=O)CCO1 c1(C(N2C3C(NC(c4csc(Cl)c4)=O)(CCC3)CC2)=O)c[nH]c2c(Cl)cccc12 CC(C)C(C(=O)NCC1CCCCN1C(C12CCC(C1)C2)=O)c1ccncc1 Cc1nsc(C(=O)NC2CCC(NC(=O)CNC(=O)CC(C)C)C2)c1N S(=O)(=O)(CC(=O)NCC12CC(CNC(=O)CCC3CCC3)(CO1)C2)NCC C1(C(=O)NCCN2CC=CC2)(COC)CCCN1C(=O)C(=O)NCC(F)F C(c1ccsc1)=CC(=O)NC(CNC(=O)C(F)C1CCCC1)C1CCC1 N1(C(C(C(C(C)C)OC)O)=O)CCC2(CCCN(C(C3CC(C)(C)C3)=O)C2)C1 c1(C(C)OC)ccncc1S(=O)(=O)N1CCN(CC2C(C(=O)OC)C2)CC1 Cc1ccc(O)cc1C(N1CC(CNC(=O)CC2CCC2)CC1C)=O c1(C(=O)NC2CCCN(C(CC(CC)(F)F)=O)C2)c[nH]c2ncnc(O)c12 c1(C(=O)NCC(CO)NC(C(c2cccnc2)OC)=O)ccc2c(c1)CC2 C#CCCCCC(=O)NCC1(O)CN(C(=O)C(C)CSCc2ccccc2)C1 N1(C(CCCOCC)=O)CCC2CCN(C(=O)CCc3cscn3)CC12 C#CCC(CO)NC(=O)C(F)CC1CN(C(C2(NC(C)=O)CCC2)=O)C1 CC1CC(NC(c2cnn(C)c2O)=O)CCN1C(c1cc(F)cc(Br)c1)=O C1(C(N(CC(CN(C(C(=Cc2cccs2)C)=O)C)O)C)=O)CCC2(CC2)C1 C(C)(C)(C(=O)OC)NC(C1C(NC(C2(COC)CC2)=O)CCC1)=O C1(C(NNC(=O)NC2CC3OC(=O)OC3C2)=O)COC2CCCCC12 CCCS(=O)(=O)CC(=O)NC1CC2C(NC(c3c(OC)ccc(Cl)c3F)=O)C2C1 C(C(C)(C)NC(N(CCOCCN(C)C)C)=O)NC1(F)CC1.C(C)(C)C C(=O)(C1=CC2C=CC(C1)C2)NCC1N(C(C2(C=C)CCC2)=O)CCC1 c1(C(c2n(CCOC)nnn2)Nc2cc(O)ccc2Cl)c(F)cc(C)cc1F CC1Cc2c(F)cccc2CN1Cc1ccn(-c2ccc(F)cc2)n1 C1(NC(c2n(CC)c(O)nc2)=O)CCCCCN(C(=O)COC2CC2)C1 N1(C(CCCC=C)=O)CCC(C(=O)NCC23CCC(CC2)OC3)CC1CC C1(c2cn(C(C)C(c3cccnc3)OCn3cnc(C#N)n3)nn2)C2CCCCC12 N1(C(C(COC)OC)=O)CC2CN(C(c3csc(SC)n3)=O)CC2C1 C(=O)(C1=CCC(C)CC1)N1CCCN(CCCCNC(C(C)CC(N)=O)=O)CC1 c1(C(=O)NCCCn2ncc(C)c2)cc(CNC(C2C(C)(C)C2(C)C)=O)nn1C c1(C(=O)NCC(CCOC)NC(CCCC#C)=O)cc2c(C)c(C)ccc2[nH]1 N1(C(C(CN(CC)CC)O)=O)CC2(C1)OCC1(C(=O)O)CC21 C1(C(=O)NCc2cc(C)oc2)CC(NC(=O)CC2CCC2)C1(C)C C(=O)(C(CO)C(C)(C)C)NCC1C2N(C(C=NOC)=O)C(CC2)C1 C=CCCCCCCNC(c1cc(F)ccc1Br)c1nnnn1C1CCCCC1 N1(C(c2n(OC)cnc2C)=O)CC=C(C(C)(C)C(=O)NCc2cscc2C)C1 CCC(CC(=O)N(CCCN(C(=O)C#CC1CCCO1)C)C)C(C)C c1(OC)ccc(NC(C2(C)CCN2C(c2ccc(C)cc2Cl)=O)=O)cc1O C1(COC(C=C(C)C)=O)CN(C(c2cccc(Br)c2C)=O)C(=O)CO1 C1(NC(=O)Cn2nnnc2C2CC2)CC(F)(F)CC1NC(c1cnsn1)=O c1(CC)ncccc1C(=O)NC1(CO)CCN(C(=O)CCc2ncc(F)cn2)C1 CC(C)(CCCNC(=O)CCC1CCCCO1)NC(=O)Cn1ncccc1=O N1(C(C(=O)NCc2ccc(Cl)cc2)C2CCSC2)CC2C3CCC(C3)C2C1 Cc1cc2c(C(N3CC(NC(c4cocn4)=O)CC34CCC4)=O)ccc(C)c2[nH]1 c1(C(N(CC(CNC(C2(COC)CCC2)=O)(C)C)C)=O)cccc(O)c1[N+](=O)[O-] c1(N2CCOCC(CNC(CCOCCOC)=O)C2)nc(Cl)nc2ncn(C)c12 CCCCC(CC)CCC(=O)NCC(C)N(C(=O)CCc1cnoc1)C N1(C(CC(c2ccccc2)N(C)C)=O)CCOC(Cc2cn(C3CCC3)nn2)C1 c1(C(N2C3C(NC(C(C)OCC#C)=O)CC(CC3)C2)=O)c(C)ccc2nsnc12 N1(CC(C2CCOCC2)=O)CCN(C(c2cn(-c3cnccn3)nn2)=O)CC1 C1(C(=O)NC2C(CNC(C3(CC)CCCO3)=O)CCC2)CN2CCC1CC2 c1(CCC(=O)NC(C(C)NC(C=CCN(C)CC)=O)C(C)C)ccc(Cl)c(F)c1 c1(OC)cc(C(=O)NC2CC(C)CN(C(c3cc(C#N)cs3)=O)C2)cc(C)n1 N12CC(C)(CO)C1=CC=CC=C2c1cc(C)c(CC#N)nccccc1 c1(Nc2cn(C)c(C(=O)NCCc3cccc(F)c3)n2)nc(Cl)ccc1F c1(C(N(C(CCNC(C(CC)=CC)=O)C)C)=O)ccc(C)c(S(=O)(=O)NC)c1 C(=O)(C(O)C(C)(C)C)N(C1CN(C(c2cnn(-c3cccc(O)c3)c2N)=O)C1)C N1(C(C2(OC)CCSC2)=O)CC2(CCC2)CC1CNC(c1cnc(F)c(C)c1)=O C1(COC)(NC(C2CC=C(C)CC2)=O)CCN(C(=O)CC2CCN(C)C2=O)CC1 N1(C(C(CC)COC)=O)CCC(C2CC2)C1C(=O)N(C1CCCC1)C c1(-n2cc(CCNC(C3C(OC(C)=O)C3)=O)nn2)cc(Cl)ccc1C c1(C(N(CCC(=O)NCC(C(C)C)CO)CCCO)=O)ccc(F)c(O)c1 N1(C(CCSCC)=O)CCC(CN(C)C(C2CC(F)(CF)C2)=O)CC1 N1(C(c2cc(C)nn2CCO)=O)C2CCC1CN(C(C1CCCC1)=O)CC2 Cc1cc(C(=O)NC2CN(C(C34CC(C3)C4)=O)C2)sc1Cl C#Cc1cn(C)nc1C(=O)NC1C2CC3C(C2)C13C(N1CCOC(C)CC1)=O c1(C(=O)NCC(CC(F)(F)F)NC(C(C)C#N)=O)cc2cccc(Br)c2o1 N1(CCC(N2CC(N(C(C(C3CCOC3)OCC)=O)C)C2)=O)CCC(O)CC1 C(C(C(F)(F)F)N1CCN(C(c2ccsc2)=O)CC1)NC(c1c(OC)nsc1)=O c1(C(N(C2CCN(C(C3COC(=O)N3C)=O)CC2)CC)=O)cccc(C(C)C)c1 c1(C(=O)NC(C(C(C)C)NC(=O)C=Cc2cscn2)C)cc(S(C)(=O)=O)co1 C(=O)(CCCCCC(=O)N(CCCN(C(=O)C=CC1CCOCC1)C)C)OCC c1(OC(C)=O)ccc(CN2CC(O)(CNC(c3cnccc3Cl)=O)C2)cc1 C(C(CC(C)C)C(=O)O[Si](C)(C)C)C1CN(OC)C1 c1(CN2C(CC(N3CCCC(CCC=C)C3)=O)CCC2)c(C)nn(CC)c1C CC1(F)CCC(C(=O)NC2CC(NC(=O)C(F)(F)c3cscn3)C2)CC1 C(Cc1ccccc1)(CCNC(=O)Cc1nccs1)NC(=O)COC(F)F C1(C)(C(N2CCN(C)C(CO)C2)=O)CN(C(=O)C2=C(Cl)CCC2)C(C)(C)C1 N1(C(C2(OC)CCCC(C)(C)C2)=O)CCC2(CC1)CC(NC(c1cocn1)=O)C2 c1(C(N2C(C)CCC(NC(C(C(C)C)CO)=O)C2)=O)ccc(F)c(F)c1F Cc1cc(C(=O)N(C2CCN(C(c3cnc(N)c(N)c3)=O)C2)C)c(C)cc1Br C1(CNC(c2c(O)ccc(C)c2)=O)CC(O)C(O)CC1C(=O)NC(C)C C(C)(C(=O)NCC(C)C(=O)NCCCC1(O)CCC1)(C1(C)CC1)OC C=C(C)CC(C(=O)NCCCC1CC1)NC(C1CN2CCC1CC2)=O c1(CC)cncc(C(=O)NCC2(C(=O)NCC3(COC)CCCC3O)CC2)c1 N1(C(c2ccc(CC(=C)F)cc2)=O)CCC2(CCCN(C(=O)CSC(=N)N)C2)C1 C(Cn1ccnn1)(C(=O)NCC1CC(C)(O)C1)NC(C(C)SC(C)C)=O C1(NC(C2N(CC)CCCC2)=O)CCN(C(=O)C(n2cc(C)cn2)C)CC1C c1(C(=O)NCC2CCCN2c2ncc(I)cn2)csc2ccncc12 C1(NC(c2cnc(OC)s2)=O)CCC(C)(CNC(=O)CCCNC(N)=O)C1 Cc1noc(C)c1CN(C)C(C1CCC(NC(=O)C(N)=O)CC1)=O C1(CCNC(CC2(C)CC2(F)Cl)=O)CCCCN1C(=O)Cn1cncn1 N1(C(C2C(C)OCC2)=O)CC=CC(C(=O)NCC2(CO)CCCCC2)C1 N1(C(c2c(C)nc(O)[nH]2)=O)CC(NC(c2ccc(C(C)C)o2)=O)CC1(C)C c1(C(N2CCCC(C(=O)Nc3cncc(Cl)c3Cl)CC2)=O)cccc2[nH]ccc12 c1(C(C)OCC)ncc(C(=O)NCCC2CN(C(C3(CC)C=CCC3)=O)C2)s1 C1(CC(=O)N(C2C(C)CC2)C)C=CC(NC(=O)C(N2CCOC2=O)C)C1 C1(NC(C(C)c2ccon2)=O)CCCC12CCN(C(c1nc(=O)n(C)[nH]1)=O)CC2 C1(CNC(C(c2ccc(Cl)s2)C)=O)C2CCC(C2)N1C(c1cnn(CCF)c1)=O C1(COC)CC(N=c2[nH]c(=NCCN3CCOCC3=O)[nH]c3c(F)cccc23)C1 C(CCC(=O)NC1CC(C)(NC(=O)CCCn2ccnc2)C1)(C(N)=O)NC(C)=O C1(C)(CCNC(CCNC(COC)=O)=O)CCN(C(C2CNC(=O)N2)=O)C1 N1(C(C(COC)(F)F)=O)CC(C2(NC(C3CC3(C)C(C)C)=O)CC2)C1 N1(C(c2cn(-c3cccnc3)nn2)=O)CCN(C(C2(F)CC=CC2)=O)CC(O)C1 c1(OC)cc(C(N2CC(NC(=O)C(N)=O)C(C)(C)C2)=O)c(OC)cc1Cl N1(C(CCOCC(C)C)=O)CCC(C(=O)N2CC(C)CC(C)(C)C2)=C(F)C1 CC1(C)C(C(=O)NC2(CNC(=O)COc3ccsn3)CC2)C1CO c1(CC(=O)N(C2CCN(C(C3(CO)CC3)=O)C2)CC)nsc2ccccc12 N1(C(c2ccc(CC)s2)=O)CCN(C(=O)Cc2n[nH]cc2Br)CC1CC N1(C(CSCC#C)=O)CC2CCC(NC(=O)CCCCOC)CC2C1 C=Cc1ccc(C(N(CCNC(C2CCCCN2CCC)=O)CC)C2CC2)cc1 N1(CCCCC2C(C)C2)CCC(NC(=O)OC(C)(C)C)CC1c1ccccc1 N1(C(C2(C)CC2(F)F)=O)Cc2ccccc2C(NC(=O)CCCC2CCCC2)C1 N1(C(C(=O)Nc2cnccc2Cl)=O)CC2CCC1C(CO)C2 c1(OCCOC)cccc(CCC(=O)NC(C)CNC(C2CCCOC2)=O)c1 C12(n3cc(C)nn3)CC(C)(C1)OC2C(=O)O.c1(C(CC)(C)N)nc(C(F)(F)F)cs1 C(=O)(CC(C)NC(=O)CC1(CN(C(=O)C(C)CSC)C)CC1)OC C12(CNC(C(C(=O)OC)(C)F)=O)CN(C(C3(C(C)C)CC3)=O)CC1CCO2 C(CO)(C(=O)NCc1cn(CC(C2CN(C3CCOC3)C2)=O)nn1)NC(N)=O CC1(C)CN(C(c2cc(F)ccc2N)=O)CCC1NC(=O)C(Cl)=CCl C1(CNC(C2(SC)CC2)=O)CCN(C(c2ccc(-c3ccccc3)o2)=O)CC1C N1(C(CCC2CCCCN(C(C(CO)OC)=O)C2)=O)CCCC2OCCC12 C(=O)(CC(C(=O)N1CCCCC(N(C(=O)CC2CC2)C)C1)c1ccccc1)OC c1(C(=O)OC)sc(CC(C)CN(C(=O)C(C)OCCc2ccccc2)C)cc1N c1(OC)ccc2c(C(=O)N(C)CC3CCCN3C(=O)C(C)NC(N)=O)cnn2c1 c1(CC(=O)NC(CNC(C2CC(F)(F)C2)=O)CO)ccc2n[nH]cc2c1 CC1(NC(c2coc(CO)c2)=O)CCCCC1C(N1CC2(CCC2)C1)=O C1(CNC(c2c(C(C)C)onc2)=O)CC2(C1)CN(C(=O)C(O)C(F)(F)F)C2 c1(OC)nccc(N(C2C3CNCC23)Cc2cccc(O)c2)n1 CC(CC(F)(F)F)(C(=O)Nc1ccc(Br)nc1F)c1ccccc1 C(=O)(C(C)(O)CC(C)C)N1CCCC(CC(=O)NC2(COC)CCCC2)C1 C(=O)(CCC(=O)C(C)(C)C)NCC(CC(NOCCCOC)=O)O C(=O)(C(CCCC(C)C)NC(=O)OC(C)(C)C)N(C1C2COCC12)CCOC C1(NC(C=CCC)=O)CC1C1CCCN(C(=O)CCCOc2cccc(F)c2)C1 N1(C(c2ccc(OCC)cc2)=O)CCN(C(C2(F)CCOC2)=O)CC1C1CC1 C1(NC(Cc2ccc(C)cc2C)=O)CCC2(CC1)CN(C(C1CCC1C)=O)C2 c1(C(=O)NCC2OCCN(C(C(=O)NCCC(N)=O)=O)C2)cnc2c(c1)CCC2 c1(C(=O)NC2(CO)CCN(C(C3C(C=C)C3)=O)CC2)ccc(C)c(C#N)c1 C(=O)(C#CC1(C)CCCO1)N(C1CCN(C(=O)C(C)(CC)CO)CC1)CCC C1(C(N(CCC(=O)OC)C2CC2)=O)CN(C(c2ccc(CO)nc2)=O)CCN1C C1(CC)C(C(=O)N(C)Cc2sccc2C)CCN1C(=O)Cc1cncnc1 C(=O)(C1CCCn2c(Br)cnc21)c1[nH]c(C)c(C(=O)OC)c1C C1(CNC(c2cnc(OC)nc2)=O)CN(C(C2C=CCCC2)=O)CCC1(F)F C=CC(C)C(C)C(=O)NC1CCC(NC(C2(F)CC2)=O)CC1 c1(C(N2CC(C(C)NC(c3cc(C4CC4)ns3)=O)C2)=O)cc(=O)cc[nH]1 N1(C(CC2N(C)CCCC2)=O)CCC2(CC1)CC2Br C1(C)(CNC(COCCCOC)=O)CN(CC(C)CC(C)C)CCO1 c1(C(N2CCC(CN(c3cc(F)ncn3)C)C2)=O)c(Br)cnn1C C12(NC(C3N(C)C(=O)NC3)=O)CCCN(C(c3coc(CO)c3)=O)CC1C2 N1(C(=O)C=C2CCN(Cc3cc(Br)ccc3Cl)CC2)C2COCC1CC(F)C2 C#Cc1cnc(C(=O)NC2CN(C(=O)CCCCC#CC)CC2C)c(C)c1 c1(C(N2CCN(C(c3c(C)cno3)=O)C(CCO)C2)=O)cncc2sccc12 N#Cc1ccc(NC(C2CNCCN2Cc2cccc(C3CC3)c2)=O)cc1Br c1(NC)c(C(=O)N(C)CC2CCN(C(C3CC34CC4)=O)C2)cc(Cl)cc1Cl C1(C(C)COc2ccccc2O)CCN(C(=O)C(n2cc(CO)nn2)C)CC1 CCC(COC)N=c1[nH]c(N(C)Cc2cc3sccc3n2C)nc2c1COC2 c1(C(=O)NCC(=O)N(CCC(C)O)C)cc(O)cc(=O)o1 c1(C(N2CC(CC)N(C(=O)C=CCN(C)C)CC2)=O)cc(OC)cc([N+](=O)[O-])c1 C1(NC(c2nnnn2C(C)(C)C)CCc2cn(C)nc2)CCC=CCC1 Cc1cc(C)c2cc(C(N3CC(N(C(=O)C(C)(C)CC#N)C)C3)=O)[nH]c2c1 C1(CNC(=O)C=CCF)C=CC(NC(=O)Cn2cccc2)C1 C#Cc1ccc(CNC(=O)CC2(CNC(C34CCCC3C4(F)F)=O)CC2)cc1 C1(NC(C(C)(C)OC)=O)C2CCN(C(c3ccccc3C3CC3)=O)CCC12 C1(NC(c2cc(CC)cc(F)c2)=O)CCC2CCN(C(c3[nH]ccc3C)=O)C1C2 CC1(C)CC(=O)C=C(c2ccc(C(=O)Nc3cnn(C4COC4)c3)cn2)C1 C1(CNC(C2N(C(Cc3cn(CC)nn3)=O)CC(F)C2)=O)OC(=O)CC1(C)C N1(CCN(CC(F)(F)F)C)CCC2(CCO2)CC1 c1(C(C(=O)NC2CCC2)N(C)CCF)c(Cl)cnn1C CC(C)CC(C(=O)N(C1CC(C)(C)C1)C)NC(C1CCOCC1)=O c1(C(=O)NC(C2CCCCCO2)C(=O)O)c(C(F)F)cccc1Cl N1(C(=O)OC)CCCC1C(=O)NCCN(C(=O)CCCC1CCCCC1)C(C)C N1(C(c2c(CC)cns2)=O)CCC2(CC1)CC2C(=O)NC1CC1C(C)(C)C c1(C(N2CCC(O)(CNC(c3cn(C)nc3Cl)=O)C2)=O)cccn2nccc12 C1(C)(C(=O)NCC2CCN(C(C=C(C)C(F)F)=O)CC2)CCCCC1C CC(C)CC(CNC(C1(C)CC1(F)Cl)=O)NC(=O)C(=O)NCC(F)F C1(C(=O)NCC)C2CC1N(C(=O)CCC1CCOC1)C2 c1(N2CC(CN(C(C(C)SCCCC)=O)C)C2)nc2ccccc2o1 c1(C(=O)NCC2(NC(CC(C)C)=O)CCOC2)c(Cl)cc(CO)cc1Cl c1(C(=O)NC2(CNC(C(C)OCC#C)=O)CC2)cnn(CC)n1 N1(Cc2ccn(C(C)(C)C)c2)CCC2CC12C CCCCC(CC)C(=O)NC(C)(CSC)C(=O)N1CCC(c2cnco2)C1 N1(C(C(C)OCC)=O)CCCN(C(C)=O)CC1.c12cccc(c1)CN2 CN1CCCC(CNC(c2occc2CNC(c2cscc2Cl)=O)=O)C1 c1(C2(C)CC2)cc(C(=O)NCC2CC2CNC(=O)CP(C)(C)=O)cc(F)c1 N1(C(C(CC)(C)C)=O)CCCC2(CCN(C(=O)C#CC3(C)CCCO3)C2)C1 N=c1nc(N(C2CCCCCC2)CCNC(c2cncs2)=O)c([N+](=O)[O-])c(Cl)[nH]1 CCC(CN(C)C)C(=O)N1CCC(CC(=O)NC(C)CF)CC1 N1(C(c2nnc(C)s2)=O)CC2CCCC(NC(C3CCc4nnnn4C3)=O)C2C1 c1(CC(=O)NC(CNC(=O)CCc2ccc[nH]2)C2CC2)cocn1 c1(OCC(=O)NCC2(F)CC(NC(C3CSC3)=O)C2)ccc2c(c1)CCCC2 C(=O)(C(C)(C)C(N)=O)N(C)Cc1ccccc1CNC(c1cn(C(F)F)cn1)=O N1(C(C2N(CC)CCOC2)=O)CCC2(CC1)CCN(C1CCNC1=O)CC2 c1(CC(C)C)cc(C(N2CCCC2CN(C)C(c2ccccc2)C)=O)n[nH]1 C1(C(C)NC(=O)COCCCN(C)C)CCCCN1C(C12CC(F)(C1)C2)=O c1(C(=O)NC2CC(CNC(c3ccn(CCC)n3)=O)C2)nccc2c1CNC2=O c1(NC(C(CC2CCC2)NC(C2CC(C)(C)OCC2)=O)=O)cccc([N+](=O)[O-])c1 c1(CCNC(=O)NC(C(CC)CCO)C)ccc2ncccc2c1 CCC(CN(C)C)C(=O)N1CC(CCNC(C2(F)CCC2)=O)C1 N1(C(c2c(C)n[nH]c2)=O)CCC(F)(CNC(=O)CN2CCCC2C)C1 c1(C(N2CC(OCCNC(Cc3c(C(C)=O)csc3)=O)C2)=O)cc(Cl)ccc1F c1(C(=O)NC)cccc(NC(C2CCCN(Cc3cccnc3N(C)C)C2)=O)c1 c1(NC(C2(C)CCCN(C(CC)=O)C2)=O)c(Br)cc(F)c(Cl)c1Br N#Cc1cc(C(=O)NCCCNC(c2coc(Cl)n2)=O)n2c1CCCC2 c1(C(=O)NCC(C)(CO)NC(c2cc(Cl)c(F)c(Cl)c2)=O)ccc2nc[nH]c2n1 CC1CN(C(=O)CC2CC3(C2)CN(C(C24CCCN(CC2)C4)=O)C3)CC1(C)CO C(=O)(C(F)CC1CC1)NCC(C)CN(C(=O)CC1(NC(C)=O)CC1)C C(=O)(C(C)(C)Cc1ccccc1)NCC(C)NC(c1c(CCC)nco1)=O N1(C(c2ccc(CC)s2)=O)CCN(C(C23CCC(C2)OC3C)=O)CCC1C C1(C(N2CCN(C3CCCC3)CC2)=O)CC(Cl)CN1 N1(c2cc(N(C)C)nc(C)n2)CCN(C(C2(O)CCOCC2)=O)C(C#N)C1 C(=O)(CC(C)P(C)(C)=O)NCc1cn(C2CCCN(C(C3CC(=C)C3)=O)C2)nn1 c1(N(C(=O)CCC2CCCC2)CC(N2CC(OC(N(C)C)=O)C2)=O)sccc1Cl c1(CCC(N2CCC(C(=O)NC(c3cn[nH]c3)C)C2)=O)ccc([N+](=O)[O-])cc1 N1(C(CCCNC(=O)NCC#C)=O)CCN(C(c2csc(C)n2)=O)C(C)C1 CN1CC(=O)N(CC(N2CCC(NC(C3(Cl)CC3(F)F)=O)C(F)C2)=O)C1=O C(=O)(CCS(C)=O)N(C1CCN(C(c2ccc(N(C)C)cc2)=O)CC1)CC C(=O)(C(O)CCC(C)C)NC(C(=O)NCC(CC=C)(C)CO)C(C)(C)O N1(CC)CCOC(C(=O)NC2(CF)CCN(C(=O)Cc3cnc(C)o3)C2)C1 c1(C(N2CC(NC(C(CC)(C)F)=O)C(O)C2)=O)cc(=O)c2ccccc2[nH]1 C1(NC(C2=C(C)CCC2)=O)CC(C2CCN(C(c3cn[nH]c3)=O)CC2)C1 C(=O)(CC(C)(C)SC)N1CC(COC)(NC(c2cn(C)nc2C(C)C)=O)C1 N1(C(Cc2ccc(C#C)cc2)=O)CCCC12CCN(C(=O)C1CC1)CC2 c1(C(=O)NCC2N(C(CCC(CC)OC)=O)CCN(C)C2)coc(S(N)(=O)=O)c1 N1(C(CC(=O)NCC#C)=O)CCC(NC(c2ccc(CO)cc2F)=O)C12CCC2 c1(C(C)C)ccc(F)c(C(=O)NC(C2CCN(C(C3CCC(=O)O3)=O)C2)C)c1 C1(F)(C(=O)NCCN(C2CC2)CC)CCN(C(=O)CC(C)F)C1 N1(C(C(C)O)=O)CCCC(C(=O)NCC2CCC(F)C2)CC1 CN1CCN(C(=O)CCN2CCCC2)CC1CNC(C1CCCS1(=O)=O)=O N1(C(=O)NC2CC(OC)C2)CCCCC12CC(C(=O)OCc1ccccc1)C2 N1(C(CCCOC)=O)CC(CNC(c2c(C(C)C)cccc2C)=O)CC(C)C1 Cc1ncc(C(=O)NC2(C(=O)NCC(F)Cl)CC2(C)C)cc1C#N Cn1ncc(Cl)c1C(=O)NCC1C2CN(C(=O)C(O)Cn3cncn3)CC12 C12(CN(C(C3(OCC)CCOC3)=O)C)CCC(F)(CC1)C2.C12(CC1)C(=O)N2 C1(NC(C2(CC#C)CCC2)=O)CC2CC1CN(C(c1ccc(CC)cc1F)=O)C2 c1(C(N2C3CN(C(C(C)Cc4ccccn4)=O)CC32)=O)cc2cccn2cn1 C1(OC)CN(C(c2cnn(C3CC3)c2)=O)CCC1NC(=O)C(C1CC(F)(F)C1)O S(=O)(=O)(c1ccc(C#N)c(NCCOC(C)C)c1)NCC(CC)(C)C C1(COC)(CNC(=O)COCC2CCC2)CCN(C(C2(C)CCC(=O)N2)=O)CC1 Cc1nnc2ccc(C(=O)NCC(C)N(C)C(C3CCOCC3)=O)cn12 CC1CN(C(=O)C(O)CCN(C)C)CC1C(N1CCC=CC1C(=O)NC(C)(C)C)=O Cc1cc(N)c(C)nc1C(=O)N(C1CCC2CN(C(=O)C3=CCSC3)CC12)C c1(C(N2CCC(N(C(c3ccnn3C(C)C)=O)CC)C2)=O)ccnnc1S C(=O)(CCCC(C)SC)N(CCNC(=O)C=Cc1cnc(C(C)(C)C)s1)CC N1(C(C2C(C(C)C)CCC(C)C2)=O)CCC(NC(=O)C(C)(F)F)C(CO)CC1 N1(C(c2n(C)cnc2)=O)CCN(C(=O)Cc2cc(F)ccc2F)CC(C)(C)C1 CC(C)S(=O)(=O)c1ccc(NC(=O)CC2(O)CCN(c3ncc(Br)cn3)CC2)cc1 C1(N(C(=O)NS(=O)(=O)C2CC2)CCNC2CCC2)CCCOC1c1ncc[nH]1 C1(NC(C(C)(C)NC(=O)NCC=C)=O)CN(C(=O)Cn2cc(Cl)cn2)CCC1C c1(CN2CC3C(C(=O)Nc4c(Cl)cc(Cl)cc4Br)(C3)C2)c[nH]c2nccc(Br)c12 N1(C(=O)C(=C2CCCCC2)F)CCC2C(CCCN2C(=O)Cc2ccns2)C1 CC1CN(C(C2CCCNC2=O)=O)CCCN1C(c1cc2ccncc2s1)=O CCN=C(NCCNC(=O)C(C)(C)C)NCC(CC(C)C)OC.OC N1(C(COCC(C)C)=O)C2CCC(C2)C1CNC(C1CC12CC(F)(F)C2)=O C(C1CCc2cc(Br)ccc21)NC(C1CC1c1ccc(F)cc1)=O N1(C(c2c(CCC)n[nH]c2)=O)CCCC(NC(=O)C(C)CC(N)=O)CC1 C1(NC(c2cc(CC)on2)=O)CCCC(N(C(=O)CC2CC2)C)C1 N1(C(C=CCC)=O)CC(NC(C2CCC(CC)CC2)=O)CC1C Cc1ncnc(C(=O)NC2(C3CN(C(C4CCCC(C)CC4)=O)C3)CC2)c1C C1(C(=O)OCC)(NC(c2cnnc(O)c2)=O)COC(C)(C)C1 c1(C(=O)NC(CC(C)NC(CC(=C=C)C)=O)C)cc2ccc(Cl)cc2c(=O)o1 S(=O)(=O)(c1ccc2nc(N3CCOC(C(N)=O)C3)ccc2c1)NCC(=C)Br CC1=NNC(=O)C1CCC(=O)NCC1CC(NC(=O)CC(C)(F)F)C1 c1(NC(CCC2(C)CN(CC3(C)NC(=O)NC3=O)C2)=O)cc2cccnn2c1 c1(C(N(CCOCCCN(C(=O)CCCCC2CC2)C)C)=O)cc(N)ccc1O c1(C(N2CCC(O)(c3cn(-c4cccnc4Cl)nn3)C2)=O)ccc(F)c(Cl)c1 c1(OC)ccc(NC(N2CCC(c3cccc(C(=O)O)c3)C2)=O)cc1S(C)(=O)=O NC1C2CCN(CC3CC(=O)N(CCC(F)(F)F)C3)CC12 C(C(C)(C)C#CC(=O)NC(CO)(CO)CO)NC(C1C(CC)C1)=O N1(C(CC(=O)NCC)=O)CCC(C)(NC(=O)C(c2ccccc2)C)CC1 C1(O)(c2cn(CCCCCN(CCN=[N+]=[N-])C)nn2)COC(C)(C)OC1 CC1(C)CC(NC(C2CC(=O)N(O)C2)=O)CCN(C(C2(C)CCCC2)=O)C1 n1(CC(C)C)ncc(C(N2CC3CCC2C3)=O)c1-c1ccccc1 N1(C(CCCN(C(C)C)C)=O)CC2COCCC2(NC(=O)CC2CCCOC2)C1 N1(C(CCCSC)=O)CCN(C2CCN(C(=O)CCC3CC3(C)C)CC2)C(=O)C1 C(C(C)CC(=O)NCCC1(C(=O)NC2C(C)C2C)CCC1)OC c1(OC)cnc(C(=O)NC(C)(CNC(c2ccccc2)=O)CC(C)C)c(OC)n1 c1(C(=O)NC(CCN(C(C(F)OC)=O)C)C(C)(C)C)ccc2nc(C)sc2c1 CCCC(CCCNC(C1(C)CC=CC1)=O)NC(c1coc(C(F)F)n1)=O c1(OC)ccc(SCC(N2CCCCC2CN(C)C(c2nocc2Cl)=O)=O)cc1 C(=O)(CC1=NNC(=O)C1)NCC1CC(NC(c2c(C)[nH]nc2Cl)=O)C1(C)C c1(C(=O)Nc2cccc(NC(C(C)NC(N)=O)=O)c2)onc2ccccc12 C1(CNC(=O)CCN(C(=O)CCC2CCC2)CCCO)C=CCCC1 N1(C(c2nccc(OC)n2)C(=O)Nc2ccc(F)cc2)CCC2(CSC2)C1 c1(-c2c(C)cco2)nc(C(=O)C(C)SC(C)C)n(Cc2ccccc2)n1 c1(CC)ncc(NC2(c3nnnn3C3CC(F)(F)C3)CCN(C3COC3)C2)cn1 c1(C(C(C)OC(C2CC(CC)C(=O)CC2)=O)=O)c[nH]c2nc(Cl)ccc12 Cc1ncc(C=CC(=O)NCC2CCN(C(c3n[nH]c(C4CC4)n3)=O)C2)c(O)n1 c1(CC(=O)NCC2CC(NC(CN(C(=O)OC)C)=O)C2)cc(OC)ccc1C C1(C(=O)NC(CC=C)C2CC2)CC(O)(CNC(C2CN(C(C)C)C2)=O)C1 C(=O)(C1=NOC2COCC12)CCN(N1C(CC(=O)NC)CC1)CC(=O)OC N1(C(CN2CCN(C)CC2)=O)CC(CNC(C2CC3(C2)CC(O)C3)=O)C2(CC2)C1 N1(C(C23C(C)OC(CC2)C3)=O)CC2(CC(NC(=O)CCc3ncccn3)CO2)C1 c1(OC)cccc(F)c1C(=O)NCCC1CC(NC(c2ncnc(O)c2Cl)=O)C1 N1(C(C2CC3C(C)(C)C3C2)=O)CC2CCC(CNC(=O)Cn3cccn3)(C2)C1 C(=O)(C1=NNC(=O)CC1)N1CCC(N(C(=O)CCC(=O)N2CCOCC2)C)C1 N1(C(C(C)OCCCCCC)=O)CCC(NC(c2c(Cl)csc2Cl)=O)CC1C C(C1CN(C(c2sccc2CC)=O)CC1C(=O)NC(Cn1cncn1)CC)=CC C(=O)(C1=CNC2=NCCC2=C1)N1CC(CCC)N(C(=O)C(O)C(C)(C)C)CC1 C1(C(=O)NCCCNC(CC(C)SC)=O)CC2C(C1)C2(C)C N1(C(Cc2nnc(C)o2)=O)CC(NC(=O)OC(C)(C)C)CC12CCOCC2 c1(C(N2CC3(CC(CC(=O)N(CCN(C)C)C)C3)C2)=O)c(Cl)cc(F)cc1Cl Cc1cccc(C(O)C(=O)NCCNC(c2ccnc(N3CCCC3)n2)=O)c1 C12(NC(c3c(C)snc3)=O)CCCN(C(c3ccnn3CC(C)C)=O)CC1C2 N1(C(c2c(C)c(F)ccc2)=O)CCOC2CN(Cc3ccc(O)c(C#N)c3)CC12 c1(-c2ccc(NC(c3cc(OC)cc(OC)c3)=O)s2)ccc2ncn(CC)c2c1 C=CCN(OC)C(=O)C1CCC(NC(=O)Cn2nnc(C)n2)C1 C1(C(=O)NC)CC(O)CN1C(=O)CC1CCC(NC(=O)C=Cc2cccnc2)C1 CN1C(=O)C(C(=O)NCC(CO)NC(C2(CC3CC3)CC2)=O)Cc2ccccc21 C1(OC)CC(C)CN(C(=O)CC(O)CNC(C2CC3(CSC3)C2)=O)C1 c1(C(=O)OC)nc[nH]c(=NCCN2CC(CNC(=O)C=CCCC(F)(F)F)C2)c1F C1(CC)CN(c2ccccc2)CCN1CC(=O)CC1CC1 c1(NC(c2nnnn2CCC2(C)CC2)(C2CC(=C)C2)C)cccc(C(N)=O)c1F C1(Br)(Cc2ccc(OCC(=O)N(CC)CC)cc2)CC12CCC2 C1(NC(C2CCC(CC)O2)=O)(CO)CCN(C(C2(OC)CCOCC2)=O)C1 N1(C(C=CC=CC)=O)CC2CN(C(=O)Cc3ccc(O)nc3)CCC12 N1(C(C(CC)N(C)C)=O)CCCCC1CNC(=O)Cn1ccc(Br)n1 CN1CCC(=O)N(C(=O)CCC2CCN(C(=O)C(C)(C)C)CC2)C1=O c1(C(N2CCC(N(c3nccc(OC)n3)C)C2)=O)cnc2n1CCOC2 N1(C(C2=CCN(C(C3(OC)CCCC3)=O)CC2)=O)CC2CCN(C)CC2C1 C=CC1(C(=O)NCCC23CC(CCO2)C3)CCN(C(=O)CC2CCC2)C1 C12(CNC(CCCNC(C)=O)=O)CC(CO1)N(C(C1(N(C)C)CCCC1)=O)C2 C(=O)(CCCC(=O)N(C)C)NCCC(=C)CNC(C1CCCCC1CC)=O CC(C)(CO)C(=O)NC1C=CCN(C(c2cnccc2C(F)(F)F)=O)C1 CC1CCc2sc(C(=O)NCCC3(NC(=O)CN(S(C)(=O)=O)C)CC3)cc2C1 C1(CN(C)C(C2(NC(c3ncccc3N)=O)CCSC2)=O)CCCCCC1 c1(C2C(C(=O)NOCCOC3CC3)C2)ccc(Br)s1 Cc1c(C(CO)NC(=O)C(C)Cc2ccccn2)cccc1Br N1(CC(C)(C)NC(C(C)O)=O)CCN(C(C2CC(=O)C2(C)C)=O)CC1 c1(CN(CC(=O)N(CC(CC)C)c2cccs2)C)nc2ccccc2c(=O)n1C C1(NC(C(COC)OC)=O)CC(CNC(=O)C(C)(C)NS(C)(=O)=O)C12CCC2 C1(CC(=O)NCC2CN(C(C34CCC(CC3)CO4)=O)CC2O)CCCC2(CC2)C1 CON(CCC(=O)N1CCCc2ccnn21)C(=O)c1ccncc1N S(=O)(=O)(c1c[nH]ccc1=NC(C)CC1CC1)NC(c1nnc2n1CCNC2=O)C c1(CNC(CC2(N(C(C(CCC)N(C)CC)=O)C)CC2)=O)cccc(C#N)c1 C1(NC(C=NOC)=O)CN(C(c2ccc(Cl)cc2F)=O)CC1C1CC1 C(=O)(CCC(C)OC)NC(CN(C(=O)COC(C)=O)CC)C.C(CC(C)C)N Cc1cc(C)c(CC(=O)NCC2(NC(C3CCCC(OCC(F)(F)F)C3)=O)CC2)s1 CCS(=O)CC(=O)N(C(C)CNC(C1CC1C(C)O)=O)C c1(Oc2ccc(C(=O)OC)nc2)ccc(C)c(NC(=O)NC2C=CC(CO)C2)c1 N1(C(c2n(C(C)C)nnc2)=O)CC(CNC(=O)C(CCO)N(C)C)C2(CCC2)C1 N=c1[nH][nH]c2ccc(C(N3CCC3CNC(c3ccc(Br)s3)=O)=O)cc12 C(=O)(C(C)(C)S(C)(=O)=O)NCC1(CNC(c2c(C)nc(CC)s2)=O)CC1(F)F C1(C)(CC(=O)N(CCCNC(c2ccnn2-c2ccncc2)=O)C)CCOCC1 c1(C(N2CC(C)C(NC(C3CC4CC4C3)=O)C2)=O)ccnc2ncccc12 C1(CNC(C2(C)C(C)C2)=O)CCCC2CN(C(c3ccc(=O)n(C)n3)=O)CC12 Cc1[nH]nc(C(=O)NCC2CC(NC(=O)Cc3ccc(Cl)nc3)C2)c1[N+](=O)[O-] C1(C(=O)NCCCCNC(CCc2ncc(C)[nH]2)=O)CCCSC1C c1(SC2CCCC(C)C2)c(F)c(F)c(C#N)c(F)c1C#N C1(CNC(c2cc(OC)nn2C)=O)C2CCCC1N(C(C1CC(C)(C)CO1)=O)C2 C1(NC(CN(CC(=O)NC(C)C)C)=O)CC(NC(C2CCCC2C)=O)CC1O c1(OC)ccc(C(N2CC(CNC(=O)CC(C)O)(OCC(F)F)C2)=O)c(OC)c1 N1(C(c2c(Br)cnc(C)n2)=O)CCC2C(CCN2C(=O)CN2C(=O)CNC2=O)C1 c1(CCCC)ccc(S(=O)(=O)NCc2ccc3nnnn3c2)cc1 CC1(C)CN(C(=O)Cc2ccc(Cl)nc2)CC1CNC(c1ccccn1)=O C1(C2(C)N=N2)CCN(C(C2(NC(C3CC(=O)C3(C)C)=O)CCOCC2)=O)CC1 Cn1cc(C=CC(N2CCOC(CNC(c3sccc3F)=O)C2)=O)cn1 C#CCC(C)(C)C(=O)N1CCN(CCN(C(=O)C(F)CC)C)CC1 C=C(C)CCC(c1nnnn1C1CCC1)NCCn1cc(Cl)cn1 N1(C(CC2(C)CN(Cc3cccc(F)n3)C2)=O)CCC2SC(=O)C=C2C1 N1(C(c2cn(CCC)nc2)=O)CCC(CNC(=O)C(C)(CC)CC)C(F)(F)C1 C1(C(N(CC#CC)C)=O)CCC(C2CC2)N1C(C1CC1F)=O C(CCCC(C)(C)NC(=O)C=Cc1ccncn1)NC(C1C(C)OCC1)=O C1(C(=O)NCC2N(C(c3cn(C)[nH]c3=N)=O)CC3(CC3)C2)CCc2n[nH]cc2C1 c1(C(=O)NC23CC(NC(c4c(C)noc4)=O)(C2)C3)ccc(CO)nc1 c1(CCC(=O)NC(CNC(CCn2c(C)ncc2)=O)CO)ccncc1Br c1(C(N(CCN(C(c2cn(CC)nn2)=O)C(C)C)C)=O)cn2ncccc2n1 N1(C(COCC)=O)CC2(CCC2NC(C2CC(=O)N(CCN(C)C)C2)=O)C1 Cc1cccc(S(=O)(=O)N2CCNC(C(N3CC4CCC(C3)O4)=O)C2)c1 c1(-c2cc(NCc3cc(OC)c(O)cc3)ncc2)cccc(S(C)(=O)=O)c1 C1(C(N2C(C(CNC(CCC(C)(C)C)=O)(C)C)CCC2)=O)CC(C(C)(C)C)=NO1 N#Cc1cncc(C(=O)NCCC(=O)NCC(F)CO)c1 c1(CC(C)NCC(=O)N(C(c2cccc(Cl)c2)C)CC)ccc(Cl)cc1 N1(C(C(C)CN(C)C)=O)CCC(NC(C23CC2C3)=O)C12CCCC2 CCCC(C)C(=O)NCCN1CCN(C(=O)CC2CC(C)=NO2)CC1 N1(C(c2cc(Cl)ncc2Cl)=O)CCC2(CC1)CCN(C(C1CCCCC1)=O)CC2 C12(CCN(C(=O)CCCCC)CC1)C(CC(C(=O)CCC(C)O)=O)N2C.CO c1(C(=O)NCCCCCCNC(CC(CC)CC)=O)cnc2[nH]nc(O)c2c1 N1(C(C(CC)(COC)CC)=O)CC(CO)C2(C1)CN(C(=O)CCNC(=O)CO)C2 c1(C(N2CCC(CCOC)(NC(=O)Cc3ccco3)C2)=O)nnn2c1CSCC2 N1(C(c2sccc2Cl)=O)CCCCC2(C1)CN(C(=O)C(c1ccc(F)cc1)F)C2 N1(C(C2CC(C)SCC2)=O)CCC2C(NC(c3cn(C)cn3)=O)C2C1 N1(C(c2cc(OCC)n[nH]2)=O)CCC(CNC(c2ccc(N)cc2)=O)C1(C)C c1(C(N2CCC(C)(NC(CCC=CC(C)C)=O)C2)=O)n[nH]c2c1COC2 C1(CC=C)(NC(=O)C(CC)CO)CCCN(C(c2cc(C)nc(O)c2)=O)C1 c1(C(=O)OC)c[nH]ccc1=NC1CN(C(=O)CSc2cnn(C)c2)CCC1C N1(C(C=CC(=Cc2cnc[nH]2)C)=O)CC(NC(c2sc(CO)nc2C)=O)C(C)C1 Cc1sc2ncc(C(N3CC(F)(F)CC3CNC(=O)CN3CC=CC3)=O)n2c1C N1(C(C2CCC(=O)NC2)=O)CCC2(CCCC2NC(=O)C(CO)C(F)(F)F)CC1 N1(C(C(=O)NCCCC2CC2(Cl)Cl)=O)CCC12CCOCC2 C(=O)(C1CCCn2cnnc21)NC1C2CCC(CN(C(CNC(C)=O)=O)C2)C1 n1(CCC)ncc(C(=O)NCC2CC(C)N(C(c3ccnc(CO)c3)=O)C2)c1C c1(C(N2C(CNC(C3C(C)C3)=O)COCC2)=O)ccc2[nH]cc(C#N)c2c1 CCCC(C)C(=O)N(CC(=O)NC1CCN(C2CC2)C1)CC(C)C C(=O)(C1=NNC(=O)CC1)N1CCCCC(NC(C(C)CC2CCCCC2)=O)C1 C1(N(C(COCCCC)=O)C)CN(C(C2(C)CCCOC2)=O)CC12CC2 N1(C(CCCSC)=O)CC2C(NC(C3CCN(C)C3=O)=O)C2C1 C1(C(N2CCCN(C(CC(CC)OC)=O)C(CO)C2)=O)CCC(C2CCC2)CC1 N1(C(C(CC)F)=O)CC(CNC(=O)Cc2ccc(C(N)=O)cc2)OC2COCC12 C1(CNC(C=CCCC)=O)C(O)C(O)CN1C(c1cc(C(C)(C)C)on1)=O c1(OC)cccc(-c2nc(C(C)NCC3CCC(=O)N3C)cs2)c1 Cc1nn(CCF)cc1NC(c1csc(C(F)(F)F)c1)=O Cc1c(C(N2CC3C(NC(C4CCCC(C)(C)O4)=O)C3C2)=O)cncc1Cl CON1CC(C(=O)NCCC2(O)CCN(C(=O)C(F)=C3CCCC3)CC2)CC1=O c1(C(=O)NC2CC3(CN(C(C(C)CF)=O)C3)C2)ccc(S(C)=O)cc1 Cn1cc(C=CC(=O)NC2CC=CCC2C(=O)NCC2CNC(=O)C2)cn1 CC1CNC12CCOCC2.C(=O)C(O)CCCc1ccccc1 C1(CC)CN(C(c2c(C)noc2C(C)C)=O)CCC1NC(=O)CN1CCCCC1 N1(C(C(C)=C(C)C)=O)CCC(CNC(=O)C(C)OC2CCOC2)C1(C)C C1(COC)(CNC(=O)CC2(C)CC2(Cl)Cl)CCCN1C(c1ccccc1O)=O c1(CSC)ccc(C(=O)NCCN(CCOCCO)C(C2COCCO2)=O)cc1 C1(OC)CC(C)CN(C(=O)COC2CN(C(=O)Cn3ccc(=O)cc3)C2)C1 C1(F)(C(=O)NCC(CNC(C(C)=C(CC)C)=O)O)CS(=O)(=O)CC12CCC2 CC(C)CCC(C)(c1nnnn1CC1CC1)NC(C)CC(F)(F)F CCCC(CCNC(C1(NC(=O)CNc2ncccn2)CC1(C)C)=O)C1CC1 C1(N(C(C2C(C)C2)=O)C)CC2CCC(C1)N2C(c1ccn(-c2ccncc2)n1)=O C1(C(=O)NC(CNC(c2ccc(C(=O)NC)nc2)=O)C)Cc2c[nH]cc2S1(=O)=O c1(C(=O)NCC2C(NC(C(C)C3CC3)=O)CC2)ccc(-c2nccs2)cc1 C(N=c1[nH]c2c(c(=NCCOc3ncccn3)[nH]1)COCC2)c1nc(Br)sc1 CC(C)CC(Cn1cc(-c2cccnc2F)nn1)NC(C1(C)COCCO1)=O C1(NC(C(C)C2CC2)=O)CCN(C(C2CCCCN2N=O)=O)CC1O C12(CNC(CC(CN)c3ccc(Br)s3)=O)CC(CO)(C1)C2(F)F c1(C(=O)NC2C(C)CN(C(c3n[nH]cc3C(F)(F)F)=O)C2)c(N)sc2c1CCC2 Cc1c(Br)cnn1CC(=O)NC(C)CCNC(c1cc(C(F)F)ccn1)=O N1(C(CC2CC(=O)C2)=O)CCCC2(CCC(NC(=O)Cn3cc(CO)nn3)C2)C1 N1(C(CC(CC)c2ccc(C)cc2)=O)CCC2(NC(c3cnsc3)=O)CCCC12 C(=O)(C1OCC(C)c2ccccc21)NCC(C)(C)NC(c1c(CCC)nco1)=O C1(O)(Cn2cc(CCC(C)O)nn2)CCN(C(c2cc(C3CCC3)no2)=O)CC1 C(C(=O)NCc1ncco1)(C(C)(C)C)NC(C(C)CC1CCCC1)=O c1(C(C(=O)NCC(C)CN(C)C(c2cnc(Cl)s2)=O)(C)C)c(F)cccc1F C1(NC(c2cccc(C)n2)=O)CCCC12CN(C(c1ccc(C)c(CO)c1)=O)C2 C12(C(N3CCC(OCCNC(C(C)O)=O)C3)=O)C3C4C1C1C2C3C41C#N c1(C(=O)NC(C(=O)N2C(C(=O)NC)CC2)Cc2ccccc2)ccccc1Br C1(CNC(Cc2nnc(C)o2)=O)(NC(c2cn(C)nn2)=O)CCCCC1C Cc1cc(F)ccc1-c1noc(C2CCCC(N)C2)n1 CC(C)CC(CNC(C1CN(C(=O)N(C)C)C1)=O)NC(c1ncccn1)=O CC1(C=CC(=O)NC2(CO)CCN(C(C34CCC(CC3)C4)=O)C2)CCOCC1 C1(C(N(C)CCNC(C2CC2Cc2ccccc2)=O)=O)CCC(C2CC2)CC1 N1(C(CCOCCOC)=O)CCCC(C)C1CNC(=O)C(C(C)C)NS(C)(=O)=O Cc1cccc(C(N2CCN(S(=O)(=O)C(Cl)(Cl)Cl)C3CC23)=O)c1[N+](=O)[O-] C1(NC(C(Cn2cccn2)NC(Cc2c(C)nsc2)=O)=O)CC2CC1C(O)C2O c1(-c2cccc(C#C)c2)ccc2nccc(C(=O)Nc3cc(C)cc(F)c3)c2c1 C1(C)(Cn2cc(C(CC)NC(=O)CCOCCCOC)nn2)CCCC1(F)F c1(C(=O)NC2(COC)CN(C(C3CCC(CC)C3)=O)C2)cc(CO)n(C)n1 C=C=C(C)CC(=O)N1CC(NC(=O)CC(C)CN(C)C)C(F)C1 n1(CC(=O)NC(CC)CNC(C2CC(N(C)C)C2)=O)ccc(=O)c([N+](=O)[O-])c1 N#Cc1ccc(O)c(C(N2CCC3(CC(NC(=O)C=CC(F)(F)F)C3)C2)=O)c1 C1(C(C)C)N(Cc2ccc(N3CCN(C)CC3)cc2Cl)CC12CCS(=O)(=O)CC2 c1(C(N2CCC(CC#C)(C(=O)N(C3CC(OC)C3)C)C2)=O)occ2c1CCC2 Cc1cc(CCC(N2CC=CC2C(=O)N(C)Cc2ocnc2C)=O)no1 c1(C(N2C(C)CC(NC(C3C(OC)CCC3)=O)C2)=O)cc2ccccn2n1 c1(C(=O)OCc2cn3cc(Cl)ccc3n2)cc(F)c2[nH]nnc2c1 N1(C(C(CCCC)O)=O)CCN(C(=O)CC(C)C(C)(C)C)CC(C)(C)C1 c1(C(=O)OC)sc(Cl)cc1S(=O)(=O)N(C(C)Cc1cccc(OC)c1)CCO N1(C(c2cn(C)nc2Br)=O)CCC2C(CCCN2C(=O)CCC(N)=O)C1 CCC(CC)C(C(=O)N1CCC(NC(C2CCN(C)C2=O)=O)C1C(C)C)OC N1(C(=O)Cc2cc(C(F)(F)F)ccn2)CCOC2(C1)CN(CCn1cccn1)C2 CCCCC(O)C(=O)NC1CCN(C(c2cc(-n3ccnc3)ccc2Cl)=O)CC1 C1(NC(C(n2c(C)ccn2)C)=O)CCCCN(C(c2nn(C)cc2N)=O)CC1 CCCCC(C(=O)NCCC1(OC)CN(C(=O)CC(F)(F)F)C1)NC(N)=O c1(C(N2CCC(C)(CNC(C3(CC#C)CC3)=O)C2)=O)cc(C(N)=O)cc(C)c1 C1(NC(C2C(COC)C2)=O)C=CCN(C(=O)C(Cc2ccccc2)NC(C)=O)C1 C=Cc1cncc(C(=O)N(C(C)CN(C)C(c2nn(C)cc2C(=O)OC)=O)C)c1 CCC(N=c1[nH]c(N2CC=CCC3(CCCC3)C2)nc(=NC)[nH]1)C1CC1(C)C C1(CNC(c2c(CC)ccs2)=O)CCC(F)(CNC(C2CC2CC(C)C)=O)CC1 Cc1cc([N+](=O)[O-])cnc1C(=O)N(C)CC1(NC(C2CC2C2CCCC2)=O)CC1 N12CCCC(C1)NC(=O)CC2.c1(C2(CCOCC)CC2)ccccc1 c1(C(=O)NC2(CF)CCN(C(CN(C3CCC3)C)=O)C2)cccc(F)c1C(F)F c1(N(C)Cc2c(C)oc(-c3ccco3)c2)nc2ccccc2s1 n1(CC)cc(Br)c(C(N2CCC(F)(CNC(=O)CC3CCC3)C2)=O)n1 CP(C)(=O)c1ccc(C(N2CC=CC(NC(c3cncc(Cl)n3)=O)C2)=O)cc1 c1(C(=O)NC(C)CCCCNC(=O)C=Cc2ccsc2)cccn2cnnc12 C1(CNC(CNC(=O)OCC=C)=O)CCCC(NC(=O)CCn2cc(C)cn2)C1 c1(C(=O)NC2C(CNC(COCC)=O)CC2)cc(Cl)cn1CC C(C(CNC(=O)Cc1cnnn1C)C(F)(F)F)NC(c1c(OC)nccc1)=O C1(C(N2CCC(C(C)NC(C3CCC4CC4C3)=O)CC2)=O)CCC(F)(F)CC1 N1(C(c2c(C)nco2)=O)CC(NC(=O)CCCCCN(C)C)C2(CC2)C1 C1(C)(CNC(C=CCN(C)CC)=O)CCCN(C(c2cnccc2C(F)(F)F)=O)C1 CC(C)C(C)CCN=c1ccc(-c2ccccc2)n[nH]1 C1(CNC2(C)CN(C(=O)OC(C)(C)C)CCO2)CCC2C(=O)NCC(=O)N2C1 CN1C(=O)CC(C(N2CCC2CNC(c2c[nH]ccc2=N)=O)=O)C1c1cnn(C)c1 c1(C(N2CCCC2C2CC2)C(=O)NCCCC)cccc(C2CCOCC2)c1 CCS(=O)(=O)CCCSc1nnc(-c2cnccn2)n1-c1ccc(F)cc1 C(=O)(CC(C)(C)C1CC1)NCC(C)CN(C(=O)C1=CCCS1)C C1(C(=O)OC)CC2(C1)CC(N=c1[nH]c(=NCCSC(C)(C)C)[nH]c3ccsc13)C2 N1(C(c2ccnc(OC)n2)=O)CC2=C(C1)CN(C(c1ccc(N(C)C)nc1)=O)C2 C=CCC(F)(F)CN(C(=O)C(C(C)O)NC(=O)CC1CC2C=CC1C2)C O(NC(=O)C(C1CCCO1)NC(=O)COCCCN=[N+]=[N-])CC(C)C#N C1(C(=O)NCCN(C(C(=CC2CCCC2)C)=O)C2CC2)CC2(C1)CC2F c1(CC(=O)NCC2(CNC(C(CC)OC)=O)CC2(F)F)csc2nccn12 CC1(C(=O)NCC2CN(C(c3ccc(C(N)=O)cn3)=O)C2)CCCS1(=O)=O C1(CNC(=O)CC2(CC=CC(=O)Nc3cc(CO)ccn3)CCC2)CCCC(O)C1 c1(OCC)ccc(CC(=O)OC2C(SCC)CC2)cc1 C(N=c1[nH]nc(-c2cccnc2)s1)C1CC(NC(C(C(C)C)N(C)C)=O)C1 CCCS(=O)(=O)CC(=O)NCC12CCC(NC(c3csc(C)n3)=O)(CO1)C2 c1(C(=O)NC2CC(CCNC(CC3(C=C)CC3)=O)C2)c(Cl)csc1Cl N1(C(C(C)N(C)CC)=O)CCC(F)(C(N2CCN(CC(=O)NCC)CC2)=O)CC1 N1(C(C(CCOC)(C)C)=O)CCC2CCN(C(c3ccn(C(C)C)n3)=O)CC2C1 c1(NCCC(C=C)(C)C)[nH]c(=NCCNS(C)(=O)=O)nc2c1ncn2C(C)C c1(C(=O)OC)ccc2c(c1)CCN(C(c1ccccc1-n1cccc1)=O)CC2 Cc1nccnc1C(N1CCCC(C(C)NC(C2CC(n3cnnc3)C2)=O)C1)=O C12(C(=O)NCC(C)CNC(=O)CC3CSC3)CCCCC(=O)N1CCC2 N1(C(c2oc(C(=O)OCC)c(C)c2)=O)CCN(C)C(CNC(=O)CCCSC)C1 C1(C(N(C(C#C)C)C2CC2)=O)CCN(S(C)(=O)=O)CC1 C(=O)(CC(F)(F)F)N(C)CC1CCN(C(C2CCC3CC23)=O)C1 c1(CC)nc2ccc(Cl)cn2c1C(=O)NCC12CC1CN(C(=O)C(C)C1CC1)C2 C1(NC(C(F)OC)=O)CN(C(c2coc(CC3CC3)n2)=O)C2CCCCC12 N1(C(c2ccc(Cl)cn2)=O)CCCC(C2CC2NC(C2(O)CC2)=O)C1 N1(C(CN(C(C)C)C)=O)CC(CNC(=O)CN2CC3CC3C2)C(C)C1 C(=O)(CC1C(=O)Nc2cc(OC)ccc21)N1C(CNC(C(C)=CC)=O)CC(O)C1 C1(CNC(c2c(NC(c3[nH]cc(C)c3)=O)ccs2)=O)CCS(=O)(=O)C1 C1(CCC(=O)NCCOCCC(C)C)CCCCN1C(=O)CCC1CCCC1 C(=O)(CCCC(C)NC(=O)C(C1CCCC1)OC)NC(CC(=O)OCC)C c1(C(N(CC(F)F)CCN(CC)CC)=O)cccc2c1OCCO2 c1(C(N2C(C)CC(CNC(COC)=O)C2)=O)ccc(C(C)C)nc1C C1(Cn2cc(-c3ccn(CC)n3)nn2)CCCN(C(c2c(Br)cnn2C)=O)CC1 c1(CNC(=O)C(F)C(F)(F)F)cnn2c1CN(C(C1(O)COC1)=O)CC2 N1(C(c2c(C)cc(Br)cc2)=O)CCC(F)(F)C(NC(c2ccc(O)c(Cl)c2)=O)C1 C1(CNC(C2C(C)C2)=O)CCCC12CCN(C(C1(C(F)F)CC(F)(F)C1)=O)CC2 C(=O)(CCCCCCSC)NC1(CC=C)CN(C(=O)CCCOCC2CC2)C1 c1(C(=O)NCCCCN(C(=O)CNC(N)=O)C)cc2sc(=O)n(C)c2s1 C1(C(N(C)CC2COCCN2C(C2C(F)(F)C23CC3)=O)=O)CCC(F)(F)CC1 CCC(C)CC(C)C=C(CNc1cc(C#N)c(Br)cn1)CC C1(NC(c2nn(C)c(Br)c2)=O)CN(C(c2ccc(O)nn2)=O)C2(CCOC2)C1 S(=O)(=O)(c1cccc(Br)c1)N1CC(CN(C)C(c2ccc(=O)oc2)=O)C1 c1(C(N(CC(N2C(CC(=O)OC)CCC2)=O)C(C)C)=O)ccc([N+](=O)[O-])[nH]1 N1(C(C(CC)CO)=O)CCCC2(CCN(C(c3ccc(O)nn3)=O)CC2)C1 CCCC(N=c1cccc(S(=O)(=O)NCC2CCSC2)[nH]1)c1ccco1 C1(CN(C(=O)OC2CCC(C(CC)(C)C)CC2)C)CC2(CCCC2)C1 c1(C(=O)OC)cc(=NC2CCCC(CNC(=O)OC(C)(C)C)C2)[nH]nc1C c1(C(N2CCC(C)(NC(C3OCCC(C)C3)=O)C2)=O)c(O)nnc2c1COCC2 CC(CC(=O)NCC1CCN(C)C1)N(C)C(c1cocn1)=O c1(C(N2CC(CC=C)(NC(=O)C(C)C(CC)CC)C2)=O)cnn2c(OC)cccc12 O=C(CCC1CCc2ccccc21)NCC1CCN1C(=O)Cc1csc(Cl)n1 c1(C(N2CCN(C(COCCC#C)=O)CC2C(F)F)=O)cccc2ccncc12 N1(C(COc2c(CC)cccc2)=O)C2CCC1C(NC(=O)C(C)C(C)C)C2 N1(C(CCC(C)SC)=O)CC2CN(C(=O)C=CC(C)(C)C)CCC12 C1(C(=O)NC(Cc2cn(CC(C=C)O)nn2)C(=O)OC)CC(C2CC2)=NO1 Cc1cc(C(=O)N(CCCN(C(=O)CC(F)(F)F)C)C)cc(N)c1O c1(C(C(=O)N2C(CNC(C3CN(C)C3)=O)CC2)(C)O)cccc2ccccc12 N1(C(c2n[nH]c(=N)[nH]2)=O)CC2CC1CN(C(=O)CC(C(F)(F)F)N1CCOCC1)C2 N1(C(c2ccc(SC)s2)=O)CC(C)CN(C(=O)COC(F)F)CC1C C(=O)(CCS(=O)(=O)C(F)(F)F)N1CC(C)N(C(C2C3COCC23)=O)CC1 Cc1nn(C)cc1S(=O)(=O)N1CCCC1CNCc1c(Br)cc(F)cc1Br c1(C(=O)NCc2c(C)ccs2)cccc(NC(c2cscc2C)=O)c1 C1(CCC)C(=O)NC(=O)C2C(=C)C2C(=O)N1.C(C)(C=CCC)C(=O)OC c1(C(N2CCC(NC(C34C(C(N)=O)(CCC3)C4)=O)C2)=O)ccc2ccoc2c1 c1(C(C)F)cccc(NC(=O)C#CCNC(C2CC2(C)C(F)F)=O)c1 c1(C(C)NC(C2(CO)CCCO2)=O)ccc2c(c1)CN(C(=O)C(N)=O)C2 C1(CCNC(=O)C=CC=C(Cl)Cl)CC(NC(=O)CNC(=O)C2CC2)C1 c1(C(=O)NCC(C2(O)CCN(C(=O)C(C3CC3)C3CC3)C2)C)ncc[nH]c1=O C(=O)(CCS(=O)(=O)C(F)(F)F)N(C1CCCN(C(c2cc(C)n(C)n2)=O)C1)CC N1(C(c2c(SCC)cccn2)=O)CCN(C(C23CC(C)C2C3)=O)CC1C c1(Nc2ccccc2)ccc(C(C)NCC(C)SCC)cc1 C(C)(C(=O)N(O)CCCN(C)C(=O)OC(C)(C)C)c1ccc(C)nc1 C1(NC(C2(C#C)CC2)=O)CN(C(C2(N3CCOCC3)CCC2)=O)CC1C CCC(CNC(C1CCN(C(=O)Cc2c(C)noc2C)C1(C)C)=O)(CC)CC C(=O)(CC(C)CC(C)(C)C)NCCCCN(C(C(C)=C(CC)C)=O)C C1(c2n(CC=C)c(C(C)SC(C)C(N3CCCCC3)=O)nn2)CCCCCCC1 c1(CC(C)C)cc(NC2CC(CNC(=O)Cc3ccc(C(F)F)cc3)C2)ncn1 N1(C(C(C=C)O)=O)CCCCC(CNC(c2cc(C)cc(C)n2)=O)C1 C1(CNC(C2C(=C)CC2)=O)CCC2(CN(C(=O)CCc3cnn(C)c3)C2)O1 CC1CN(C(c2c[nH]c(=N)s2)=O)CC(C)N(C(c2c[nH]nc2OCC(F)F)=O)C1 n1(CC)ccc(C(=O)N(C2CCN(C(c3cnoc3CC(=O)OC)=O)C2)C)c1C Cc1ccc(C(=O)NCC(C)N(C(=O)C(c2ncccc2F)(F)F)C)cc1CO c1(OC)nc(N2CCCC(CNC(C3CC(C(C)C)C3)=O)CC2)nc2[nH]cnc12 C1(OC)CCC(CC(N2CC(NC(c3c(C(F)F)cnn3C)=O)C2)=O)CC1 C1(CNC(C2N(C(CCC)=O)CCC2)=O)CCCN(C(C2CCCC2(C)C)=O)C1 C1(CC)CCN(C(=O)Cc2cncc(C)c2)C(CNC(c2cnn(C)c2Cl)=O)C1 c1(OCC(CC)NC(c2ccc(=O)n(CCO)c2)=O)ccc2c(c1)CCC2 C1(F)(CNC(Cc2cc(C)sc2)=O)CCN(C(=O)C=Cc2ccc[nH]2)C1 N1(C(Cn2c(C)c(Cl)cn2)=O)CC(NC(c2nnc(O)cc2O)=O)C(C2CC2)C1 N1(C(c2c(SC)csc2)=O)CCC2CN(C(c3cncc(C)c3)=O)CC2C1 C1(NC(c2cccc(O)c2Br)=O)CC2(C1)CC(NC(C1CCCO1)=O)C2 C1(CC(N2CCC(O)(CN(C(c3c(C)onc3)=O)C)C2)=O)CC2CCC(C1)C2 c1(CN(C2(CC)CNC2)C(c2cc(CC)ncn2)=O)c[nH]c2cccc(Cl)c12 C1(CCC)CCOCC1(c1nnnn1C(C)(C)CC)NCc1ccc(CC)nc1 O=NN1CCCCC1C(=O)NCC1CCC(F)(CNC(=O)COCC(F)F)CC1 C1C(=O)NNC1=O.c1(OC)ccc(-c2nn(-c3ccccc3)c(=O)n2C)cc1 C1(CNC(C(CC)C(F)(F)F)=O)CN(C(=O)CCC(C)(C)F)CCC12CCC2 c1(SCC(=O)NCC2N(C(C(C)C3CC3)=O)CCC2)ccc(Cl)cc1Cl C1(C(=O)NC(C)C(C)C(=O)NCC2(C)CCCCO2)C2CCC(C2)C1C C1(NC(C(CC)(C)CO)=O)CN(C(=O)Cc2ccc(Cl)cc2F)CC(F)(F)C1 C1(CC)(CC)CC(NC(C2(C)COC(=O)OC2)=O)CN1C(=O)Cc1ccnn1C C=CC(C)CC(=O)NC(C1CCCCC1)CNC(C1(COC)CCCC1)=O c1(C(=O)NCCN2CCN(C(C3C(=C)C3)=O)CC2)cnc2c(C)cnn2c1 c1(NC(c2ccc(-n3cccn3)cc2)c2cc(OCC)ns2)cnc(OC)nc1 c1(C(=O)NCC2(NC(c3sc(C)cc3C)=O)CC(OC)C2)ccc2c[nH]nc2c1 c1(OC)ccc2c(c1)CC(C(=O)NNC(=O)C13CC(c4ccccc4)C1C3)O2 C1(NC(c2nnnn2-c2ccc(F)cc2)CCOC)Cc2ccccc2C1C c1(C(N2CCCC(N(C(CC=CC=C)=O)C)C2)=O)nc(N2CCCC2)nc(=N)[nH]1 Cc1ncnc(NCCCOC(c2cccc(OCCN(C)C)c2)=O)c1Br CC1CCN(C(c2cccc(CNC(=O)CC3CC4CC4C3)n2)=O)C1CO N1(C(C(CNC(C(C)(C(C)C)OC)=O)O)=O)CC2CCC(C1)C2C#N CC(C(=O)NC(c1ccccc1F)CNC(=O)Cn1nccn1)S(C)(=O)=O C1(CNC(CCCN(C)N=O)=O)CN(C(C2SCCS2)=O)CCC12CCOC2 c1(C(=O)NCCN(C2CCCC2)C(C2C(CCC)C2)=O)cc2c(nc1N)CCCC2 c1(OC)cc(C)c(C(=O)N(C)CCN(C(=O)CC(=O)NC2CC2)C(C)C)cc1Cl C(C1=CCN(C(C2CC(CNC(C3(CO)CC=CCC3)=O)C2)=O)CC1)OC C(C)(C)(CC(=O)NCC1CNC(=O)CO1)N(C(CCCC)=O)C C#CC1CN(C(=O)C(C)N(C(c2cn(C(C)C)nn2)=O)CC)CCN1C c1(C(N2CCC3(CCCN3C(c3scnc3Cl)=O)C2)=O)cnc2c(c1)COCC2 CCCCC(C(=O)NC1CC(CNC(c2cn3ccsc3n2)=O)C(O)C1)N(C)C c1(CNC(C2(NC(C3N(C)CC(O)CC3)=O)CCSC2)=O)cn2ccccc2n1 C1(NC(c2csc(Cl)n2)=O)(CO)CCN(C(=O)C=CC2CCCCC2)C1 Cc1noc2nc(C(N3CC4(CC4)CC3CNC(c3coc(O)n3)=O)=O)ccc12 CC1C(C)N(C(C2C3CCC2(c2ccco2)C3)=O)CCN1C(C1CCNC1=O)=O C1(NC(C2CCC(C)(C)CC2)=O)CN(C(=O)C(N)=O)C2CCCCC12 c1(C(=O)OCC)ccc(CCc2ncoc2CNCC2CC(O)C2(C)C)cc1 N#CCCCC(=O)NC(CCC1CCC1)C(=O)NCc1cccc(CO)c1 C1(CNC(CCSC)=O)CCN(C(C2CCCN(CC(F)F)C2)=O)C1(C)C n1(C(CC)C)nnnc1C(c1cncn1CC)NCCCCF C(C)(c1cccnc1)=CC(=O)NC(CNC(c1cc(OC)n(C)n1)=O)C1CCC1 c1(C(=O)NCCC(=O)NCCCOCC)snc(C)c1N c1(C(=O)OCC)cc2n(c1)CCN(C(c1cccc(OC3CCCC3)n1)=O)C2 c1(C(N2C(NC(c3cnn[nH]3)=O)CCC2)=O)ccc(S(=O)(=O)NCC2CC2)cc1 Cn1ncc(CNC(C2(C)CC2(C)C)=O)c1C(=O)NCc1c[nH]nc1C1CC1 C1(CC(=O)NC2CC(CNC(c3ncc(OCC)nc3)=O)C2)OCCCC1(C)C c1(C(N2C(CNC(C(C=C)(C)C)=O)CC3CC32)=O)ccc2[nH]c(=O)c(=O)[nH]c2c1 Cn1cnc(N2CCCC2C2(NC(C3CC3c3ccccc3)=O)CC2)cc1=O c1(CC)c(C(=O)NC(C)(CNC(=O)COCP(C)(C)=O)C2CCC2)cccc1F CC1CN(C(C2(CO)CC=CC2)=O)CC1CNC(=O)OC(C)(C)C CC1CN(c2nc(C3CCCC3)ns2)CC1NC(=O)C(=O)NCC(F)F C1(CCC(=O)NC2CC(NC(CNC(=O)NCC3CC3)=O)C2)CCCOC1 N1(C(C(C2CC2)OCC)=O)CCCN(C(=O)COC2CCOCC2)C(C)C1 c1(OC)ccc2c(c1)C(C(=O)NCCCCCNC(=O)C(F)CC(C)C)CCC2 C(C(CC1CCCC1)C(=O)N1CCCCC1CCO)NC(c1cnc(C)o1)=O N1(C(C(CCC)C#N)=O)CC(C)(C)CCC1CNC(C1CC(F)(CO)C1)=O c1(OC)ccccc1CC(=O)N(CCCN(C)C(C1C2CCCC12)=O)C CC(C(F)(F)C(F)(F)F)=CC(=O)NC(CNC(=O)CCCC(=O)N(C)C)C1CC1 N1(S(CC)(=O)=O)CCCCC1C(=O)NC1C2CCN(C(c3cccnn3)=O)C12 C1(C(CNC(C2CC2(C)C(F)F)=O)NC(C2(C)CC2)=O)CCCCC1 C1(C)(C(=O)NC(CCC)C2CC2)CN(C(c2ncn(C(C)C)n2)=O)C(C)(C)C1 c1(CSC)ccc(C(=O)N(CCCNC(=O)Cc2cccc(C3CC3)c2)C)cc1 Cc1nn(CC#N)c(C)c1NC(=O)Nc1ccc(Br)cc1CCCN C1(CC)C(C(=O)NCc2ccn(C(C)C)n2)CCN1C(=O)CN(C)C(N)=O N1(C(C2COCC(C)(C)O2)=O)CCC(C2(NC(c3ccc(O)nn3)=O)CC2)C1 c1(NCC2CCCN(CC)C2)nccc(=NCCc2cc(C)on2)[nH]1 N1(C(c2c(C)oc(C(C)C)n2)=O)CCC(NC(=O)C(C)N2CCC2)CC1C n1(C2CC(OCC)C2)c(N2CCC(C3(C(N)=O)CC3)CC2)nnc1C1CCOC1 C(=O)(CS(=O)(=O)CC(=O)N1CCc2sc(CNC(=O)C(O)C3CC3)nc2C1)OC CC1=C(C(=O)NC(C)CNC(c2ccc(S(C)=O)cc2)=O)C=C2CCCN=C2N1 C(C(=O)N1CCSC(C)CC1)(C(C)(C)C)n1cc(C(C(C)C)O)nn1 CC1CCCN(C(C2CC(CF)C2)=O)C1CNC(=O)CC1(C2CC2)CC1 N1(C(C(C)OCC(C)C)=O)CCC(CCC(=O)NCCOCCOC)C1 C1(NC(c2cccc(N(C)C)c2)=O)CC2CC(NC(C3CCN(C)C3=O)=O)C2C1 N1(C(C=C(C)I)=O)CCN(CCO)CC1.C(=O)C(F)C1CCC1 c1(OC)ccc(-c2cn(CCOc3ccccc3Cl)nn2)cn1.C1CN(C)CCN1 C#Cc1ccc(CNC(c2ccc(-c3nccc(OCC)c3OC)nn2)=O)cc1 CC(O)C(C(=O)NCCC(C)NC(C1CC1(Cl)Cl)=O)N(C)C(=O)OC(C)(C)C C1(CC(=O)NCCC(C)NC(c2ccc(C3CC3)cn2)=O)COC(C)(C)C1 S(=O)(=O)(c1ccc(S(=O)(=O)NCc2cccc(F)c2Cl)cc1)N(c1ccno1)C N1(C(c2n(CC)c(O)nc2)=O)CC(F)(F)CC1CNC(c1ccnc(C)c1)=O CC1CC=C(C(=O)NCC(CNC(C2(C)SCCCS2)=O)CO)CC1 C(=O)(C1=CCCN(C(=O)Cn2cccnc2=O)C1)NCC(C)(C)C#N C1(CNC(C(C2CCOC2)OCC)=O)C(C)CCN1C(C1CCC(C)C1)=O CC1CN(C(c2ccc(CN=[N+]=[N-])cc2)=O)CCC1NC(C1(C)CC1(F)Cl)=O C1CNCC1c1cn(-c2ccsc2C)nn1.COCOC(C)C C(=O)(C(CNC(C1(O)CC1)=O)N(C)C)NCCN(C)CCF N1(C(c2n(C)ccn2)=O)CC2C(C(=O)NC3CCCC(OC)C3)C2C1 N1(C(Cc2c(F)ccc(OC)c2)=O)CC2CCN(C(=O)CCCCOC)C2C1 c1(NCC(CC)(C)F)nc(N2CCN(C(=O)C(C)O)CC2)nc2c1ncn2C C(=O)(C(CC)C(C)C)NCc1cn(CC2N(C(CCCCC)=O)CCC2)nn1 C1(NC(CCN(c2ccccc2)C)=O)CN(C(C2(CCF)CC2)=O)CCC1F c1(OC)cnc(Br)cc1C(N1CCC(O)(CNC(=O)C(C)(C)CO)C1)=O CC(CC(=O)NCC(c1ccccc1)NC(=O)CN(c1ccccc1)C)C(F)F CC(CC(=O)NCC(C1CCC1)NC(c1cc(N)ccc1F)=O)C(F)F C=CCC(CC(=O)NCC1(CF)CC1)NC(C1CCCC12CCC2)=O Cc1ccccc1CCCNC(=O)Cc1noc(C(F)(F)F)n1 C(C)(C(C)CCCCC(=O)O)NC(c1cc(C)c(-n2cnnn2)cc1)=O N1(C(C(=O)NCC)=O)CCC2(CCC(CNC(c3cn(C)nn3)=O)O2)CC1 c1(C(N2C(C(C)NC(CC)=O)CCC2)=O)ccc(-c2ccc[nH]2)cc1 C1(CNC(C2C(=C)C2)=O)CCCN(C(c2ccc(-n3cccn3)cc2)=O)C1 Cc1nc(C(=O)NCC2CC(CNC(C3CCC(O)C3)=O)C2)nn1-c1nc[nH]n1 N1(c2ncc(OC)cn2)CCC2(CC2C(=O)Nc2cc(SC)ncn2)C1 c1(C(=O)NCC(C2CCCC2)NC(C2C(C)C2)=O)sccc1S(C)(=O)=O Cc1nncc(CNC(C2CCOCCN2C(=O)CC2CC3CC3C2)=O)c1C C1(NC(c2ccc(Cn3ccnc3)o2)=O)COCCN(C(=O)C(O)CC(F)F)C1 C(N=c1[nH]cnc2c1SCCC2)C1C(NC(C(C(C)C(F)(F)F)F)=O)CCCC1 N12CCCC(CC1)NC(=O)C2=O.C1(C(CC)NC(=O)CNC(=O)NC)CCCO1 CON(CCC(=O)NC(C)C=CC(N1CCCC1)=O)C(=O)CC(Cl)Cl N1(C(C2(NC(C3CCN(C)C3)=O)CCC2)=O)CCCC(CCC(N)=O)C1 N1(C(c2cncc(C)c2Cl)=O)CCC2(CCN(C(=O)CCc3cnco3)CC2)C1 N1(C(c2c(C)snc2)=O)CCN(C(C2CC2C2CC2)=O)CC1CC(C)(C)C C(c1ccc(F)cc1)=CCC(=O)NCC1(CNC(C(C=CCCC)O)=O)CC1 Cc1cc(C(=O)N(C2CCCCC2)C(c2ccco2)C)c(Br)c(Cl)c1 C1(C2CCC2)(CNC(CC(CC)C(F)F)=O)CCN(C(=O)C(F)(F)C(C)O)CC1 c1(CN(CCC(C)CCO)c2nnnn2C2CCCCC2)cc(F)ccc1F c1(NC)cncc(C(N2CCOCC2CNC(C2CC2CC(C)(C)C)=O)=O)n1 C1(CNC(c2cc(C)c(C)s2)=O)CCN(C(=O)C2=CCCS2)CC1C CC1CC=C(C(=O)NC2CC(NC(c3ccc(OC(F)(F)F)c(Cl)c3)=O)C2)CC1 N1(C(CCCCOC)=O)CCC(C2CC(NC(c3sc(C)cc3Cl)=O)C2)C1 N1(C(c2c(C)nc(Nc3nncs3)s2)=O)CCCC(C(=O)NCC(C)C)CC1 c1(C(=O)NC2CC(NC(C=Cc3cc(C)no3)=O)C(O)C2)c(F)ccc(C)c1F C(=O)(CCCCC(=O)OC)NC(CC)C(=O)N1CC(COC)C1 Cc1nn(C)cc1CC(=O)NC(CCN(C(=O)CCC1CC(F)(F)C1)C)C(C)C Cc1cc(C(=O)NCCc2c(F)cc(Br)cc2F)nc2[nH]nc(O)c12 CC1CN(C(=O)OC(C)(C)C)CC(CC2(C(N3CC4CN(C)CC34)=O)CC2)O1 C1(COC)(NC(C2CCC(C)S2)=O)CCN(C(=O)CCCC(N)=O)CC1 c1(OC)ccc(CC(=O)NCC2(C)CCN(C(=O)CCCC#N)CC2)cc1OC C1(C)(COC)CC2=C(C(=O)N1)C(c1c(C)n(C)nc1C)NC(=O)N2CCC#N c1(C(=O)NCC(C)(C)NC(=O)CC2CCCC23CC3)cc2c(Cl)cccc2[nH]1 CCC(C)C(C(=O)NCC1CCCCCC1)N(C)C(c1nccs1)=O c1(CCC)ccc(C(=O)NCC(C)(C(C)C)NC(C2CCC2C)=O)cc1 C1(N(C)C(C2C=CCCC2)=O)CCCCC1NC(=O)C(C)(C)C1CCCC1 C12(C(=O)NC3C(C)N(C(C4CCCC(C)C4)=O)CC3)CC3CC(C1)C(=O)C(C3)C2 N1(C(c2nccc(CC)c2)=O)CCC(NC(=O)C(N2CCNC2=O)C)C(O)C1 C1(C(N(CC#C)CCOC)=O)(CC)CCCN1C(=O)C(C1CCOCC1)C C1(CC(=O)NCC(C)NC(=O)CCC2OCCO2)CCCOCC1 c1(C(=O)NC(CC=C)CNC(=O)C(C)(C)NS(C)(=O)=O)nn(C)c(Br)c1C CC(O)(Cc1ccccc1)C(=O)NC1CN(C(c2cnccn2)=O)CC1O Cc1cc(OCC(=O)NCCCNC(=O)C(F)C(C)(F)F)cc(C)c1Cl n1(C2(CC(=O)N(C(C)CNC3(CC#C)CC3)C)CC2)ccnc1 C1(NC(c2ncc(OC)nc2OC)=O)CCN(C(c2cnc[nH]2)=O)CC1(C)C CC1(C)CC(C(N2CCCC3(CC2)CC3)=O)CN(C(c2ccc(O)nc2)=O)C1 c1(-c2ccc(CNCCCN3CCC(O)CC3)s2)cc(F)cc(Br)c1 Cc1ccc(-c2cn(C3CN(C(C4(F)CCOC4C)=O)C3)nn2)cn1 CC(C)(C#N)CC(=O)NCCN(C(c1ccc(C#N)cn1)=O)CC1CC1 c1(OC)ccccc1CC(N1CCSC2CC12)=O c1(C(N2CCC(O)(CNC(C3(OC)CCCCC3)=O)C2)=O)cc(C)c(C)cc1C C(CCC(=O)N(CC(C)(C)CNC(=O)CC1(C)CCCO1)C)OCCOC C(C)(C)(CCCN=c1[nH]c2ccccc2s1)NC(CC1C(C)C1)=O Cc1cc(NC(C2CC(F)CN(C(=O)CN3CCOCC3)C2)=O)cc(F)n1 N1(C(CNC(C)=O)=O)CCCC1C1CCCN1C(=O)CNc1ncccn1 C1(CCC)CCCCN1C(C1CC12CC(NC(C1C3CCC(F)C13)=O)C2)=O N1(C(c2ccc(C)c(CO)c2)=O)CC(C)(C)OCC1CNC(=O)C(C)CN(C)C CC1=C(C(=O)N2CCCC2(C)C(N2CCC(F)(CO)C2)=O)CC1 c1(C(N2CC(C)(NC(c3cnc(C(F)(F)F)s3)=O)C2)=O)cnn2c1OCC(O)C2 N1(C(C(c2cccs2)SC)=O)C2CCC1C(NC(c1cc(F)ccc1Cl)=O)C2 CCCC(CC)CCC(=O)N1CC(C(=O)Nc2c(C)cc(C)cc2C)C(C)(C)C1 C1(Nc2cc(NC(C)CS(N)(=O)=O)ncn2)CCOC2(CCOCC2)C1 N1(CCC#C)CCC(C(=O)NC(C)C(CO)NC(C2(CC#C)CCCC2)=O)CC1 N1(C(CCCc2onc(C)n2)=O)CC(NC(c2sncc2C)=O)C(C)(C)C1 C1(COC)(NC(=O)C(C)=C2CCCC2)CCCN(C(C2CCC(C)O2)=O)C1 C1(NC(C(C(C)C)F)=O)CC12CCC(NC(C1CCC(N(C)C)CC1)=O)CC2 CCCCC(C)(C)C1(n2ccnn2)CC1.n1(CCC=O)cc(C2CCCC2O)nn1 N1(C(C(c2n(C)c(Br)cn2)(F)F)=O)CCC2(CO)CCCC12 c1(CN(C(C)C)C(=O)NC(c2cc(Br)no2)C)ccc(C(F)(F)F)cc1 CCC(CC)C(CCN=c1nc2scnc2c(NCC(C)CC(=O)NC)[nH]1)OC Cc1ccc(F)c(C(N2CCN(C(=O)C(C)N3CCCC3)C(CF)C2)=O)c1 C(C)(C)(CCC(=O)NC(CNC(C1(c2cc[nH]n2)CC1)=O)C(C)C(C)C)OC c1(C(N2C3C(CNC(c4scc(OC)c4)=O)C(C3)C2)=O)cc2cccnc2o1 N1(C(C2CC(C)(CC)C2)=O)CCCCC2(CCN(C(=O)C(C)(C3CC3)OC)C2)C1 Cc1cc(O)cc(C)c1C(N1CC(CCNC(c2ccc[nH]2)=O)OC(C)C1)=O N1(C(CCc2scc(C)n2)=O)CCC2CCC(C1)N2C(C1(F)CCC(C)CC1)=O C(N=c1[nH]c(Cl)nc2cc(C)sc12)C1C(C(F)(F)F)CN(C(C(CC)(C)OC)=O)C1 c1(C(=O)OC)cccc2c1CCOC2C(=O)N1CCC2C(CCCN2C)C1 c1(C2(C)CN(C(=O)NCc3ccnc(F)c3)C2)ccc(F)c(F)c1 Cc1nc(C)c(C(N2CC(NC(C3(C)CC3(F)F)=O)CC(F)C2)=O)nc1C C1(C)(CC)C=C(C(=O)NC2CC(NC(c3cc(OC)ns3)=O)C(O)C2)C1 C1(C)(CNC(c2n(CC#C)cnn2)=O)CC(F)(F)CN1C(C1CC(O)C1)=O Cc1cc(C(=O)NCC2CCC(C)CN2C(C2CC(F)(CO)C2)=O)cc(O)n1 C(=O)(CS(=O)(=O)C1CCCC1)NC1CC(F)(CNC(C(C)NC(N)=O)=O)C1 CC1=CCC(CCC(N2CC3CC2(c2cn(-c4ccc(C)nc4)nn2)C3)=O)CC1 C1(CNC(C(C)S(C)(=O)=O)=O)CCCC12CCN(C(C1(C)CC=CCC1)=O)CC2 C1(C(N)=O)CN(C(=O)Cc2cc(C3CC3)no2)CCC1NC(=O)CC1CC1 C1(F)(CNC(C2ON=C(C)C2)=O)CCN(C(=O)CC(C)(C)O)CC1 C1(NC(CCc2c(C)noc2Cl)=O)CC(O)CN(C(=O)CCc2ncccn2)C1 c1(CN2CCC(C(N(CCC(C)C)C)=O)C2)ccc(F)cn1 C(=O)(C(F)(F)C(F)(F)F)NCCC1CC(NC(c2c(C(C)(C)C)n[nH]c2)=O)C1 CCC(CC)(CCC(=O)N1CCN(C(=O)CCC(C)(C)OC)CC1)[N+](=O)[O-] N1(C(C=CC(=O)OCC)=O)CCC2(NC(c3cc(C)ccc3Cl)=O)CC2C1 CCCC(C)(CC)C(=O)NCC(C)NC(=O)C(CC(C)C)NC(=O)OC(C)(C)C C12(CNC(c3ccn(C)n3)=O)CN(C(=O)CC3CCCCC3O)CC(F)(C1)C2 C=CCC(=O)NCCCN(CCO)C(C1CC(C(F)F)C1)=O N1(C(c2c(C)ccc(C)n2)=O)CC2CCC(NC(C3CCCN3N=O)=O)CC2C1 Cc1nc(O)c(C(=O)NCCN(CCON)C(c2nonc2N)=O)nc1C c1(CC)c[nH]c(C(=O)NC2(CNC(C3CC(C(C)C)C3)=O)CCC2)n1 N1(C(Cn2c(C)nnn2)=O)CC(O)C(O)C1CNC(C1(C)CC(C)(C)C1)=O N1(C(C(C(CC)C)NC(c2cncnc2C)=O)=O)CCC2CC1C(=O)N2C c1(C(=O)NCC2C(NC(c3cccc(CCO)c3)=O)CC2)cc2ccncc2s1 C12(CNC(C(C3CC3)OCC)=O)CCCC1N(C(c1csc(Cl)c1)=O)CC2 c1(C(N(C2CN(C(C(CC#C)C)=O)C2)C)=O)cc2cc(F)ccc2o1 OCC(CN=c1[nH]c(=NCCCc2ccco2)[nH]c2cc[nH]c12)c1ccccc1 C(=O)(CC(CC)C(C)C)N1CC(CCC)C(C(=O)NCC2(OCCO)CCC2)C1 S(=O)(=O)(c1cccc(C(=O)O)c1)Nc1c(OCCCOCC)cccc1 Cc1cc2nccnc2cc1C(N1CC(NC(c2ccc(S(C)(=O)=O)[nH]2)=O)C1)=O c1(SCC(=O)NCC(C2CC2)NC(C2(C)CC(C)(C)C2)=O)ccsc1[N+](=O)[O-] CCCC(CC)C(=O)NC(CC(=O)NCC(O)CC(=O)OC)C1CC1 C1(NC(C(COC)N(C)C)=O)CCN(C(c2csc([N+](=O)[O-])c2)=O)C1(C)C N1(Cc2c(OCC)c(Br)cc(C)c2)CCc2[nH]nc(C(=O)NCC(F)(F)F)c2C1 c1(CNC(c2ccnn2C2CCCOC2)=O)nc(CSc2ccccc2)no1 c1(CC(=O)NCCCN(C(=O)CCc2cncnc2)C2CCCC2)cccc(F)c1 c1(C(N2CC(C)N(C(=O)Cc3cncnc3)CCC2)=O)cc(F)cc2nn[nH]c12 C1(NC(CCNC(=O)NC)=O)CCOCC1NC(C1(CO)CC(F)(F)C1)=O C1(CC(OC)OC(=O)OC)(C(=O)NC2CC2OC)CCCC1 N1(C(C(C(C)C)OC)=O)CC(CNC(C2CC3(C2)CC(F)(F)C3)=O)CC(C)(C)C1 C(=O)(C(CCOCCO)CCN)C(CN(C)C)=O.N1(CC(=O)NC)CCSCC1 Cc1ccc(C)c(CNC(=O)CC2CN(C(C3CCCCC3O)=O)CC2C)c1 CC1CC1C1CC1C(N1CCCC1Cn1cc(CNC(C2CCCO2)=O)nn1)=O c1(NC(C2CCC(NC(C3CN(C)C(=O)C3)=O)CC2)=O)c(C#N)cnn1C N1(C(c2ccc(COC)cc2)C(=O)NCCC)CCN(C)CC1C C12(C(N3C(C)CCC3)=O)CCCC1CCN2C(C1CC(C)(O)C1)=O c1(C(N2CCCC(C(=O)NCc3cc(Br)cs3)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 N1(C(CCOC(C)=O)=O)CC2CC(NC(c3ccc(C(F)(F)F)c(C)c3)=O)C1C2 N1(C(C2OCC(C)(C)C2)=O)CC(C)(C(=O)NCCCF)CC1(C)C c1(C(N2C3CN(C(c4ccc(F)cc4Br)=O)CC2C3)=O)cc(F)c(Br)cc1Cl Cc1ccccc1CC(N1CCCCC1CCNC(C1CC2CC2C1)=O)=O N1(C(C(=O)OC)CSc2ccncc2Br)CCc2ccccc21 Cc1nc(C)c(C(=O)NC2(C)CCN(C(C3C(c4nc(=N)[nH][nH]4)C3(C)C)=O)C2)[nH]1 c1(N2CCC(N(C(C(C)OCC)=O)C)C2)nc(C)nc(O)c1C c1(N(CCCSC)C)nc(=N)nc(N2CCCC(c3nc(C)c(C)[nH]3)C2)[nH]1 C(=O)(C(C)C1CCCO1)NC1(CCNC(CSCCC)=O)CC1 C1(C(=O)NC2C(CN(C)C)CCC2)CC(O)CN1C(=O)Cc1ccon1 C1(NC(C2(OC)CC2)=O)CCC(CC(=O)NCc2nnc(CO)s2)C1 C1(NC(=O)C(c2ccc(O)cc2)C2CC2)COCCN(C(c2ccns2)=O)C1 Cc1ccc2cc(C(N3CCC(NC(C4CC(=O)NC4(C)C)=O)C3C)=O)cn2c1 C1(C(N)=O)(CNC(=O)CCC2CCCCO2)CN(C(c2csnc2Cl)=O)C1 c1(C(N(C2CCN(C(CC(CCC)O)=O)C2)CCC)=O)cc2cc(Cl)ccc2o1 N1(C(c2c(OCC)n[nH]c2)=O)CCC2(CC1)CCN(C(=O)C(C)CN(C)C)C2 c1(C(=O)NC2CN(C(c3cn(CCC)nn3)=O)C(C)C2)cc(C)c2[nH]nnc2c1 c1(C(N2CCC(C(=O)NCC3(OC)CCC3)O2)=O)ccc2nccn2c1 N(C(=NCCc1ncccc1C)N(C)CCC1CCOC1)CC(=O)NC(C)C S(=O)(=O)(c1cccc2cccnc12)NC1(C2CC2)CC1.CC12CCN(CC1)C2=O C(=O)(C1CCc2c[nH]nc21)OC(C(C)C)CCc1ccccc1 C1(CC=C)(NC(c2nc(C)ccc2F)=O)CC2CCC(C1)N2C(=O)C(C)(F)F Cc1nc(C)n(CC(=O)NCC2CC(O)CN2C(=O)CN2CC(C)(C)C2)n1 CN=c1[nH]cc(C(=O)NC2CC2CNC(c2cc(C3CC3)nn2C)=O)o1 N1(C(CC(C=C)(C)O)=O)CCC(C)(C)C(CNC(=O)CCCCCc2cccs2)C1 C(CO)(C(C)NC(=O)COC1CCCOC1)NC(CNC(CCC)=O)=O Cc1ccc(S(N)(=O)=O)cc1NC(c1nn(-c2ccccc2)cc1Br)=O c1(C(=O)NC(C)C(=O)NCC2C=CCOC2)nn(C)cc1Cl C1(C(=O)NCC(C#C)(C)C)CN(C(c2n[nH]cc2C)=O)CC1C1CC1 CC(C(=O)N(CC(=O)NCC(C)(C)N1CCCC1)CC1CC1)n1ccnc1 N1(C(c2ncn(CC)n2)=O)CCC(C)(CNC(=O)C(N2CCC(O)CC2)C)CC1 C1(CNC(c2cn(CCC)nc2)=O)C(C)CCN1C(=O)CNC(C)=O C#Cc1cc(C(=O)NC(C)CCNC(c2ccc(Cl)c(O)c2N)=O)cc(Br)c1 c1(C(N2CCC(n3ncc(NC(C(C)S)=O)c3)CC2)=O)cccc2nc[nH]c12 C1(CN(C(=O)CCc2ccsc2)CC)CCCN1C(=O)CCc1nc(C)no1 C1(OCC)CN(C(=O)C(C)NC(N)=O)CC1CNC(c1cnnn1C)=O N1(C(C(C)CS(C)=O)=O)CCN(C(c2cc([N+](=O)[O-])ccc2N)=O)CC(C)(F)C1 C(c1cc(C)cc(C)c1)=CC(=O)NC(CCCNC(CC1N(CC)CCC1)=O)C C1(NC(c2ccc(C(F)(F)F)cn2)=O)C2CC1N(C(C1CCOC1)=O)C2 C1(C(=O)NC2CN(C(c3cn(CC)nc3)=O)C2)C2CCC(C2)C1(C)C c1(C(N2CCC(N(C)C(c3cnccc3Cl)=O)CC2)=O)ccc(S(N)(=O)=O)s1 Cc1cc(C(=O)NCC2CCC2NC(c2coc(Cl)n2)=O)cc2c1NCCC2 CCC1=NOC(C(=O)NC2CCC2C(=O)NCCCc2n[nH]c(C)n2)C1 c1(CC(=O)NC(CNC(C2OCCN(C(C)C)C2)=O)C)cc(F)cc(Br)c1 c1(C(N2CC(N(C(c3cn(CCOC)nc3)=O)C)C2)=O)cc(F)ccc1Br N1(C(CSC)=O)C2CCC1CC(CCNC(=O)CCn1ccc(C)n1)C2 CC(Cc1cccn1C)N=c1cc[nH]cc1S(=O)(=O)NCc1c(F)cccc1Cl Cc1nc2cc(C(N3CCN(C(=O)CN4C(=O)CCC4=O)CC3CO)=O)[nH]c2s1 C1(C(N2CC(=C(CNC(=O)CCCc3ccccc3)F)C2)=O)CC2(CCC2)CO1 N1(C(C2C(C)CCS2)=O)CCOC2(C1)CN(C(c1cn(C3CCC3)nn1)=O)C2 C1(C(=O)NCCOCCNC(c2cncc(O)c2Cl)=O)CCc2ncncc2C1 c1(C(N2CCC(C)(CNC(=O)C(F)=CCCF)CC2)=O)cccc2[nH]nc(O)c12 C(CCCCCNC(C1CCOC1(C)C(F)(F)F)=O)NC(C1CN(C(C)=O)C1)=O Cc1cc(Cl)ncc1CC(=O)N(C1CCN(C(=O)CCC2(C)CCC(=O)N2)C1)C C1(CC(=O)NCC(O)CNC(c2ncccc2O)=O)SC2=NCCN2C1=O CCCCC(C(=O)NC1CCC12CN(C(=O)Cc1nc([N+](=O)[O-])n[nH]1)C2)C(C)C C1(c2nnnn2CCOCCO)(NCCc2c(C)cncn2)CCC2CCCC2C1 C=CCC(C(=O)NCC1(CNC(C2(NC(C)=O)CCC2)=O)CC1(F)F)OC c1(C(=O)NCC)cnc2ccncc2c1.CCC1C(=O)N(CCOCCO)CCN1 c1(C(=O)NC2CN(C(=O)CCOc3cccnc3)CC2O)nnn2c1CSCC2 C1(N(C(C(C)OCCCC)=O)CC)CCN(C(=O)CNS(N)(=O)=O)C1 CC(C)(O)C(F)C(=O)N1CCCC(CO)(CNC(c2cnc(C3CC3)[nH]2)=O)C1 O=C(CCCCC(F)(F)F)NC1CC(NC(C2CCC(CN(C)C)O2)=O)C1 c1(C(N2CCC(C(N(CCCSC)C)=O)C23CC3)=O)cnn2ccc(Cl)c(F)c12 c1(CC)nn(C)cc1C(=O)N(CCNC(C1CCCNC1=O)=O)CCOC CC1CN(C(=O)C(F)(F)C2CCOCC2)CCC1NC(c1cccc(F)c1F)=O c1(C(=O)NC2C(CNC(C(C)(C)OC)=O)C2)ccc(C(F)F)c(Cl)c1 C(=O)(N=c1cc[nH]cc1Cl)C1CC(C)CN1C(=O)CN1CCC(C)CC1 c1(OC)ncc(Cl)c(C(N2CCC(C)(NC(=O)C(C)CSC)CC2)=O)c1Cl N1(C(CC2CC(C)C2)=O)CC(N=[N+]=[N-])CC1C(=O)NCCC1=CCCCCC1 CCC(C)C(C)C(=O)NC1CCN(C(=O)COC2(C(F)(F)F)COC2)CC1 C(c1ccccc1C)=CC(N1C(CC)C(C(=O)NCC2CCC2)CC1)=O CC(C)(C(=O)N1CC(S(C)(=O)=O)C1)C1=CCN(C(C2CC(N=[N+]=[N-])C2)=O)C1 C(=O)(CC(=O)NC1(CO)CN(C(=O)CC(O)C2CCCC2)C1)OC(C)(C)C c1(C(=O)Nc2cn(C)c(C(=O)Nc3cnc(Cl)cc3I)c2)cccc(F)c1O N1(C(C(CC)(C)O)=O)C(C(=O)Nc2ccc(Cl)c(Cl)c2)C2CC(F)C1C2 S(=O)(=O)(c1cnn(-c2ccc(Cl)cc2)c1C)N1C(C(CC)O)CC1 c1(C(=O)NCCCCNC(CN(c2ccccc2)C)=O)cc2n(c1)CCC2 c1(OC)cc(CCC(=O)NCCC(F)Cn2cc(CN3CCOC3=O)nn2)on1 N1(C(C(OC)OC)=O)CCN2CCN(C(=O)CN3CCCC3=O)CC2C1 CCCC(O)(CCC)CC(=O)N1CC2(CCN(C(c3nc(O)cs3)=O)C2)C1 N1(C(C2C(C(=O)OCC)C2)=O)CC2CC(Oc3ccsc3)C2C1 c1(CCC)cc(C(=O)NC2CC3C(NC(=O)COCC)C3C2)c(C)o1 C1(C(N(CC(CN(C)C(c2ccc(C#N)s2)=O)O)C)=O)CCn2cncc2C1 C(=O)(C1=CCN(C(C2CC23CCOCC3)=O)CC1)NCC1(C)C=CCCC1 C1(NC(C(C)(C)C2CC2)=O)CCN(C(=O)C=C(C2CC2)C2CC2)CC1F C1(C(=O)NC(CNC(Cc2cc(OC)cc(Cl)c2)=O)CO)CCC2C(C1)C2(F)F C1(C(=O)O)CN(C)CCN1C(NCOC(C(c1ccccc1)C)=O)=O.N(C)C c1(C(C)NC(C(c2cnccn2)C)=O)ccc(CNC(=O)Cn2cnnc2)cc1 C1(O)(C(CNC(=O)N(c2ccccc2Cl)CC2CCOC2)O)CCCCC1 c1(CN(C(c2cc(C(C)C)[nH]n2)C(=O)NC2CCC2)C)cn2ccccc2n1 c1(CC)nc(C)ccc1NC(c1nnnn1CC(F)F)c1ncc[nH]1 c1(C(=O)NCC(CNC(C(CC=C)C)=O)CO)cnc(O)cc1OC c1(CC(=O)NC(C)(CNC(C2COCCO2)=O)C2CCC2)ccc(F)c(F)c1 C1(CCC=C)(C(N2CCCC2C2(CO)CC2)=O)CN(C(=O)C(C)=CC(C)(C)C)C1 c1(C(c2n(C3(C)CC3)nnn2)NCc2cccc(C)c2F)c2c(nn1C)CCC2 Cc1ccc(O)c(C(N2CCC(NC(c3sncc3Br)=O)C2)=O)c1 N1(C(C)=O)CCCCC(C2CN(C(C34CC(CO3)C4)=O)C2)CCC1.c1(CC=O)nn(C)cc1Cl C(C#CCCO)NC(CN(C(=O)CC1CCC(=O)C1)CCOC)=O C(N=c1[nH]c2c(c(=NC(C)C(C)C3CCC3)[nH]1)CSC2)c1ccc(OCC)cc1 C1(C(=O)NCC2CCN(C(=O)C=CC(=O)N(C)C)C2)(SC)CC(O)C1 c1(C(=O)NC2CCCC2CC(C2CN(C3CCOC3)C2)=O)cccc(F)c1Cl c1(C(C)N)ccc(C(F)(F)F)cc1.C(C)(C)(C)OC(N(CCCCO)C(=O)N)=O c1(C(=O)NC2CCN(C(=O)CCOCC3CCCO3)C2)ccncc1Cl C(=O)(C(CC(C)CC)NC(=O)C(C)NC(=O)C1CC1)NCC(NOCC)=O c1(C(=O)NC(CN(C(=O)CC2CCSC2)CC)(CO)CO)cc2ccccc2o1 N1(C(c2cc(SC)oc2C)=O)CC2CCC(C1)N2C(=O)C=CC1CCOC1 N1(c2nnc(C(N)=O)s2)CCCC2CN(C(c3cnc(Cl)c(Cl)c3)=O)CCC12 C1(CN(CCCOC)C)CC2CN(C(=O)OC(C)(C)C)CC12 C#CCC(CC(F)F)C(=O)N1CCC(C(=O)NCC2CC(O)CC(O)C2)C12CC2 C(=O)(C(C)(C)CCS(C)(=O)=O)N1CC2C(NC(c3ccc(CC)s3)=O)(C2)C1 c1(CNS(C)(=O)=O)ccc(CN2CCN(C(c3cc(O)n(C)n3)=O)CC2)cc1 CC1(NC(C2CC2c2ccccc2Cl)=O)CCN(C(c2cccnc2O)=O)C1 C(=O)(C(C#N)C(C)(C)C)N(C(C(=O)NCCC(CCC#C)O)CC(C)C)C C(CCCCNC(=O)COCc1ccccc1)NC(C=CC(=O)OCC)=O C(=O)(CCCCC)NCCCCNC(CC=CC)=O C1(OC)(NC(=O)NC(C)CC(N2CCCOCC2)=O)CCOCC1 C1(NCc2ccc(Oc3cccc(Cl)c3)nc2)CC2CNCC(C1)C2 C1(CNC(CCCCC#C)=O)CCC2(CN(C(=O)CCC(C)SC)C2)O1 C1(NCCC(=O)NCC(C2(O)CN(C(c3cnn[nH]3)=O)C2)(C)C)CCCCC1 C1(C(=O)NC2(CN(C(c3ncc(OC)nc3)=O)C)CC2)CC2CCCCN2C1 C12(CC)CCCCN1C(=O)N(CCC1CCOC1)C2=O c1(C(N2C(C)(CNC(c3n(C=C)ncc3)=O)CCC2)=O)cc(F)ccc1C(C)=O N1(C(C2(OC)CCSC2)=O)CC2CCC(NC(=O)CSc3nnnn3C)(C2)C1 Cc1onc(C2CC2)c1C(=O)NCC1CN(C(=O)CC2CCCC2(F)F)CCO1 O=C(O)CCCS(=O)c1sccc1C(=O)OCCSN1CCCCC1.C1CO1 C1(CC(N2C(C(C)C)COCC2)=O)CC2(C1)CN(C(C1C3COCC13)=O)C2 c1(CC(C(=O)NC2CCN(C(Cc3cc(C)[nH]n3)=O)C2C)O)cc(Cl)cc(Cl)c1 N1(C(c2n(CC=C)ccc2)=O)CC(NC(c2csc(Cl)c2)=O)C(C2CC2)C1 C(=O)(C1=C(F)CN(C(=O)CC2(C)CC2)CC1)N(CC(O)C(F)(F)F)C N1(C(C(C(C)(C)C)O)=O)CCn2cnc(-c3ccc(F)cc3C(F)(F)F)c2C1 c1(CC)ccoc1C(=O)NC1(C)CC(NC(C2CC2c2ccc(C)o2)=O)C1 N1(C(C(C)CF)=O)CCN(C(c2ccc(F)c(CO)c2)=O)C(CO)C1 C12(C(C)NC(C3C(NC(CCNC(=O)OC)=O)CC3)=O)CCC(CC1)C2 C(=O)(CC1=Cc2ccccc2C1)N(C1CCN(C(C2CC(S(N)(=O)=O)C2)=O)C1)C c1(C(N2C(CN(C(c3[nH]cc(C)c3)=O)C)CCCC2)=O)cn2cccc(Cl)c2n1 C(CC(C(=O)NC1CC1)NC(=O)C(C)c1ccsc1)SC C(=O)(CCC1=CCCCC1)NC(CC=C)CNC(=O)C(=O)N(C)C c1(C(N2CC=CC(NC(C=C(C)C)=O)C2)=O)cnc2sc(C)nc2c1 C1(F)(CNC(C2=C(C)CCC2)=O)COCCN(C(=O)CCC2NC(=O)NC2=O)C1 c1(-c2c(-c3n(CCOCC=C)ccn3)n(C)nc2)cc(C)ccc1CO CN1CCCC1C=CC(=O)NC1CC(O)(CNC(=O)CCN2CCOCC2)C1 C(c1ccc[nH]1)=CC(=O)NC1(CCCNC(c2cccnc2)=O)CC1 c1(NC(C2(CCNC(CCCC)=O)CC2)=O)cccc(NC(N)=O)c1 N1(C(Cn2ncc(C)c2)=O)CC2ON=C(CNC(=O)CC(C)(C)C(C)(F)F)C2C1 c1(C(=O)NC(CCC)C(=O)NCC(O)Cn2cccn2)ncc(C)cc1C N1(CCN(C)C(c2ccsc2Cl)=O)CCN(C(=O)CC2CCC(=O)N2C)CC1 C1(C(F)(F)F)(OC)CC(CNC(c2cc(C)c[nH]2)=O)(NC(=O)CC2CCCC2)C1 N1(C(=O)C=Cc2c(F)ccc(Cl)c2F)CC23CCCC2(COC3)C1 c1(CN(CCC)CC2(OC)CCOC2)ccc([N+](=O)[O-])cc1COC C1(F)CCCCC1.N1(C(CCNC(COC)=O)=O)CCCC1C1C(C)C1 c1(OC)cc(CC(=O)NCC(C(C)C)NC(c2cocn2)=O)cc(C(F)(F)F)c1 C1(C(=O)NC(c2ncc(C)cn2)C)CN(C(=O)CC(C)(C)C#N)CC(C)(C)C1 C1(c2ccccc2)(CNc2c(C)ccs2)CCN(C(=O)Oc2ccccn2)CC1 Cc1cncc(CCC(=O)NCC(C)NC(=O)C(C)(C)CN(C)C)c1 c1(CC(=O)N(C2CN(C(c3cc(C4(C)CC4)n[nH]3)=O)C2)C)csc(NC=O)n1 Cn1nccc1C(F)=CC(=O)OCC(c1cccc(I)c1)=O C(CCCCC(=O)NCC1CC(F)CN1C(c1cncc(F)c1C)=O)=CC C1(COC)(NC(c2csnc2C)=O)CCCN(C(c2nc(=O)n(C)[nH]2)=O)C1 N1(C(c2ncc(C)c(C)c2)=O)CCCN(C(c2occ3c2CCC3)=O)C(C)C1 c1(C(N(C2CC(NC(C(CC)OC)=O)C2)C)=O)cc(OC)c(Cl)cc1Cl C(Cc1ccco1)(C(=O)NC1(CO)CC1)NC(=O)CCc1cncs1 C1(NC(c2n[nH]c(C)c2Cl)=O)CN(C(=O)CC2NC(=O)NC2=O)CCC1(C)C C1(NC(CC2N(C(C)=O)CCC2)=O)CC2C1CCN2C(c1cc(C#N)cs1)=O Cc1nc2ncccc2cc1CCC(=O)NCC#CCNC(=O)C=CS(C)=O c1(C2N(C(CC3(NC(=O)NC4CC4)CCOC3)=O)CCC2)nnc2n1CCC2 CC1CCN(C(C2(C3CCCCO3)CCC2)=O)CC1NC(c1ccc(C2CC2)o1)=O C(=O)(C1=CC2(CCOC2)C1)N1CCC2(CN(C(C(c3cnn(C)c3)C)=O)C2)C1 N1(C(C2C(F)(C(=O)OC)C2)=O)CCC(NC(c2sc(C)c(C)c2C)=O)C(O)C1 c1(C(C)NC(C(C)NC(=O)NC)=O)ccc(CNC(=O)C(F)=C(C)C)cc1 c1(-c2sc3c(c2)CN(C(Cc2ccc(C)nc2)=O)CC3)ccccc1S(C)(=O)=O N1(C(Cc2ccc(C)cc2)=O)CC2CC1CN2C(C1(C2CCCO2)CCC1)=O CCCCC(CNC(=O)CC(C)(C)OC)NC(=O)CSc1nncs1 C(CCCC(C)NC(c1sc(C)cc1OC)=O)NC(c1cnc(C(C)=O)s1)=O C(COC(C)C)(C(=O)Nn1ccccc1=O)NC(C(C=C)C)=O C(CCC(C)C(=O)N1CCC(C)(CNC(C2CCCN2C(=O)N(C)C)=O)C1)OC c1(C(N2CCCC(NC(=O)CCCN3CCOCC3)C2)=O)cnc2c(c1)COC2 N1(C(c2c(C)c[nH]c2)=O)CC2(CC(C(=O)NCC3(C)CCCCO3)CO2)C1 CCCC(C(=O)OC)C(=O)NC1CCCN(C(c2ccc(C)s2)=O)C1 c1(C(=O)NC2CCCN(C(C3(C)CCNC3=O)=O)C2)nccc(Br)c1O C1(OCC)CN(Cc2ccc(Cl)s2)CC1NC(=O)NC(C)C c1(C(N(CC(C)N(C)C(C2CC(F)C2)=O)C)=O)cc2c(nn1)CCC2 c1(C(=O)NC(Cn2cncn2)C(=O)N2CCC(CO)C2)cc(Cl)cs1 Cc1cc(Br)cc(Cl)c1NC(=O)CC1CCC(NC(=O)CC2CCCC2)CC1 Cc1oc(C(=O)N(C)CC2CCCN(C(c3cccnn3)=O)C2)cc1S(C)(=O)=O c1(C(=O)NCC(C)(CNC(=O)CSc2nncs2)OC)cnnc(C)c1 c1(N2CCC(NC(CS(CC)=O)=O)C(F)C2)ncnc2sc(C(C)C)cc12 C1(N(C(C2(c3ccccc3)CCC2)=O)CC)CCN(C(C23CC(F)(C2)C3)=O)CC1 N1(C(C2C(c3ccn(C)n3)C2)=O)CC2CC(NC(=O)CCS(N)(=O)=O)C(C2)C1 C(=O)(CCCC(=O)NCCNS(=O)(=O)NCC1CC1)N(CCCC(C)C)C N1(C(C(C)n2ccnc2)=O)CCN(C(c2ccccc2)=O)C(c2cn[nH]c2)C1 CCCCCCCCOCC(=O)NCC1(F)CC(NC(c2ccncn2)=O)C1 c1(CC(=O)NC2C(C)CCN(C(COCC)=O)C2CC)nccc2ccccc12 CC(C)(CNC(=O)CSC(F)F)NC(C1CC1c1cn[nH]c1)=O C12(CNC(Cn3cc(-c4c(OC)cccn4)nn3)=O)CCCCC1C2(F)F C(=O)(CC(C)C(C)C)N(CCNC(COc1ccc(SC)cc1)=O)C1CC1 CON1CCC(CC(=O)NCC(C2CC2)NC(C2CC2C2CCCO2)=O)CC1 S(=O)(=O)(C1(C)CC1C)NC1CC(SC)C1 c1(CC)n[nH]c(=NC2CN(C(c3cc4c([nH]3)CCC4)=O)CC(C)(C)C2)o1 C1(C(C)NC(CNC(C(C)ONC(=O)OC2CC2(F)F)=O)=O)CC2(CCC2)C1.O C(C(C)(C)C(F)(F)F)NC(C1N(C(c2cc(C)c(C)o2)=O)CC(O)C1)=O N1(C(CN(C)C(N)=O)=O)CC(O)CC1CC(N1CCC1n1cccn1)=O C(=O)(C(CNC(C12CCCC1C2(F)F)=O)CC=C)N1CCC(=CCC)C1 N1(C(C(C)=C(C)C)=O)CCN(C(C2CC(O)(c3ccccc3)C2)=O)C(C(F)F)C1 c1(OC)c(NC(=O)C(=O)Nc2ccnn2-c2cccnn2)cc(Cl)cc1Cl C1(NC(c2nc(CC)sc2)=O)CC2CCC(C1F)N2C(C1COCCN1CC)=O C1(C(=O)NCC2C(CNC(=O)C=CCN3CCCC3)C2)CC2(CCC2)CO1 C(C(CC(C)C)C(=O)N1CC2C(C1)C2(F)F)NC(c1nc(C)n(C)c1)=O c1(CC)ncc(Cl)c(C(=O)NCC(C(C)C)NC(c2ccsc2C(F)(F)F)=O)n1 c1(CC)cnc(C(=O)NCCN(C(=O)CS(=O)(=O)N(C)C)CC(C)(C)C)nc1 c1(NC(=O)C(N2CCNC3CC23)c2ccccc2)ccnc(-c2ccc(F)cc2)c1 N1(C(C(C)C(F)F)=O)CCOC2CCN(C(c3cnn(CCO)c3)=O)CC12 c1(CN2CC(CCn3cc(C(=O)OC)nn3)C2)c[nH]c2c(C)cccc12 CC(CC(=O)N1CCCCCC1CNC(c1cncc2c[nH]nc12)=O)C(F)(F)F C1(C(=O)N(C(C)C(=O)NC)C)(NC(CN(CC)CC)=O)CCSC1 CC(C)(C)C(C#N)C(=O)N1CCN(C(=O)CSc2ccccc2)CC1C1CCC1 N(C1CCc2ccc(Cl)cc21)C(C12CC(C(=O)Nc3ccccc3O)(C1)C2)=O c1(C(=O)N(C2CCCC2)CCNC(c2n[nH]cc2C(F)(F)F)=O)cn(CCF)nn1 c1(SC)ccc(C(=O)NC2CN(C(=O)C(C)(C)CO)CC2C)cc1[N+](=O)[O-] C(c1nc2ccccc2s1)=CC(=O)N(C1CC(NC(C(C)(C)SC)=O)C1)C Cc1cc(C(=O)NCCCOCCN(C(=O)CN2CC3CC3C2)C)c(N)c(C)c1 c1(CC(=O)NC(C)CCCNC(=O)Cc2nccs2)ccc(C#N)cc1F c1(C(=O)NC2CC(C)(NC(COC)=O)C2)cnn(C)c1C(F)F C1(C(N(C)CC2(CNC(CCC=C(C)C)=O)CC2)=O)CC(C)(C)OC1(C)C N1(C(C2CCC(C)O2)=O)CCCC(CNC(=O)C(c2ccc(F)cc2)C)C1 N1(C(C=CC=CC)=O)CC=CC1(C)C(N1CC(c2ccon2)C1)=O CCC(O)CC(=O)N1CCC(C)C1CNC(c1ccnc(OC)c1)=O C1(C)(CN(C(=O)CCCn2cc(-c3ccc(F)c(F)c3)nn2)C)CCCCC1O c1(OC)cc(=NC(=O)C(C)(C)CN(C)C(c2cnsc2)=O)[nH]n1C S(=O)(=O)(C1CC2(C1)CC1(CCC1)C2)Nc1cnn(C)c1-c1ccccc1 Cc1cnn(CC(=O)NC(C2CC(NC(c3cscc3Cl)=O)C2)C)c1 c1(C(N2CCC(C)C(NC(=O)CC3(O)CCC3)C2C)=O)cn(C)c(=O)n(C)c1=O N1(C(Cc2c(C)ncnc2C)=O)CCN(C(c2cc(N)c(F)cn2)=O)CC12CC2 C1(NC(C2(CC(C)C)CC2)=O)CCN(C(=O)CCCc2ccccn2)CC1F C(=O)(C1CCCc2n[nH]cc21)N(CCCNC(C1N(CCC)CCCC1)=O)C c1(OC)cc(C(N2CCN(CCCNC(c3ccon3)=O)CC2)=O)cc(Cl)c1O Cc1nc(C(N2CCOC(C(C)NC(=O)Cc3cnnn3C)C2)=O)c(C)n1C CC1(C)OCC2CC12C(=O)NCC1CN(C(C2CC2c2ccccc2Cl)=O)C1 c1(NCCCN2CCC(C)CC2)[nH]c(=NC(C)C2CCOC2)nc2c1ncn2C C1(C(C)C)CN(C(=O)CCc2c[nH]c(=N)[nH]2)CCN1C(=O)Cc1cccnc1Cl C1(NC(=O)Cc2ccc(C3CC3)cc2)CCCCC1NC(C1CSCC(=O)N1)=O CCC(O)C(C)C(=O)N1CCC(CCC2CCCN2C(=O)C(C)C(O)CC)CC1 C(=O)(CCC(=O)N1CCC(CNC(c2nnn(C)n2)=O)(OC)C1)NC C(=O)(C1CCCn2c(COC(c3c(F)cccc3Br)=O)nnc21)NCC C1(NC(N2CCC(CCF)C2)=O)CCCN(c2ccc(F)c(F)c2)C1=O C1(C(C(=O)NCCCF)N(CC(C)C)CCC#N)CC2C=CC1C2 c1(-c2cn(CC3C(CNC(C(CC)COC)=O)C3(F)F)nn2)cc(C)cnc1F N1(C(CCS(C)=O)=O)CCC(n2cccn2)(C(=O)NCC2CCCCCC2)CC1 C1(NC(c2onc(C(C)(C)C)n2)=O)CCCN(C(c2n[nH]cc2[N+](=O)[O-])=O)CC1 Cc1cc(Br)ccc1CNC(=O)CNC(=NCC1CC1C)NCC1CCCO1 c1(C(N(C)CCNC(=O)Cc2ccccc2Br)=O)ccc(-n2cccn2)nc1 c1(C(=O)NCC2C(NC(c3cnc(CC)s3)=O)CCCC2)cc(C#N)ccc1C Cc1cc(F)ccc1C(N1CCCC(C)C1CNC(C1(C#N)CCOCC1)=O)=O C1(C(=O)Nc2ccc(C(C)NC(=O)N(C)C)cc2)Cc2nccnc2C1 N1(C(CN(CC)CC)=O)CCCC(CC)C1C(N1CC2CCC2(OC)C1)=O N1(C(c2ncc(C)nc2)=O)CC(NC(=O)CCCS(C)(=O)=O)C2CCCC12 C1(C(=O)NC2CN(C(C3(CC(C)C)CCCC3)=O)CC2F)CCCCC1(F)F N1(C(c2c(CC)ccc(Br)c2)=O)CCC(C)N(C(C2CC2(C)C)=O)CC1 CC1CCc2[nH]c(C(=O)NCCC3CN(C(=O)CN4CC=CC4)C3)cc2C1 CC1CN(C(=O)C(C)(C)c2cnn(C)c2)CC1NC(c1cc(C2CC2)ncn1)=O C1(CNC(c2c(CC)nn[nH]2)=O)CCC(F)(CNC(=O)C(C)n2cncn2)CC1 c1(CC(=O)N(C2CCN(C(c3cnn(CC(F)(F)F)n3)=O)C2)C)ccc(O)cc1 Cn1cc(C(N2CCCC(c3nncn3C3CC3)C2)=O)c(-c2ccnn2C)n1 c1(OC)cnc2nc(NC(c3ccc4nn[nH]c4c3)=O)sc2c1 C1(CC=C)(NC(=O)C(C)SC(C)C)CCN(C(=O)CN2CCCC2=O)CC1 c1(NCc2ccc(CC(C(=O)O)F)cc2)cc(Cl)ncc1F N1(C(C2(F)CN(C(c3cc(C(C)C)[nH]n3)=O)C2)=O)CC2CN(C)CC2(C)C1 C1(NC(Cn2c(C)nnn2)=O)CCC2CN(C(C3CCCC(=O)N3)=O)CCC2C1 N1(C(C(CN(CC)CC)F)=O)CCN(C(c2cnc(O)o2)=O)CC1 C(CC(C)C)(C(=O)N1CC(c2cn(-n3ccccc3=O)nn2)(N(C)C)C1)OC Cc1nc2cc(C(=O)NCCCCN(C(=O)CSC(F)F)C)c(F)cc2[nH]1 Cc1ccc2c(c1)CC(C(=O)NC1(CNC(C3C4CCC(=O)C34)=O)CCCC1)S2 C1(C(N(CC(=O)NCC2OCCC2C)CCC)=O)CCCCNC1=O N1(C(C(C)(C)N(C)C)=O)CCCC(CNC(=O)C(F)C(C)(C)O)CC1 C1(CC(C)C)COCCN1C(=O)CC1CCN(Cc2ccc(-c3nccs3)cc2)C1 C1(CNC(=O)CCC2(O)CCC2)CN(C(C2(CO)CCC2)=O)CCCO1 c1(C(=O)OC)cc(NC(N(C(CC#C)C)C)=O)ncc1C c1(CC(N2CC(N(C(=O)Cc3cn(C)nn3)C)C(O)C2)=O)cccc2[nH]ncc12 c1(C(=O)NCC2(NC(C(C)OC(C)(C)C)=O)CCOC2)cnn2c1OCCC2 c1(C(C)C)ccc(C(=O)N(C2CN(C(C3CNC(=O)N3)=O)C2)C)cc1 Cc1ccc2[nH]c(CN3CC4CN(C(c5ccnc(Cl)c5C)=O)CC34)cc2c1 C(=O)(C1Cc2c(Cl)cccc21)N1CCN(C(CSCc2[nH]c(=N)sc2)=O)CC1 N1(C(c2cc(COC)on2)C(=O)NCCOC)CC(C)SC(C)C1 N1(C(c2c(CNC(C3(CC)CNC(=O)C3)=O)cc[nH]2)=O)CCCC(O)(CO)CC1 C=CC(CCC)CC(=O)NC(C)(CC)CCNC(c1ncc(Br)cc1O)=O C1(N(C(C2C(=C)C2)=O)C)CCCCN(C(c2ccc(C(C)C)c(Cl)c2)=O)C1 C(=O)(C1CCc2ccccc21)NCc1nccc(C(=O)NCCn2ncnn2)c1 N1(Cc2ncc(C)o2)CCC(NC(c2ccn(C)n2)=O)C(O)C1 C=C=CCCC(=O)NC1CCOCC1NC(C1CC1C(C)(F)F)=O CCC(C(=O)N1CCC(CN(C(c2cncc(NC)n2)=O)CC)C1)C(F)(F)F O=C1CCC(C(N2CCN(CC(=O)NCC34CCCC3CCO4)CC2)=O)CCO1 CCCC(C(=O)OC(C)(C)C)S(=O)(=O)N1CCN(Cc2ccccc2)CC1C#N CCCC(C)C(=O)N(CCCNC(c1cccc(=O)o1)=O)CC1CCCC1 CC(CN=c1[nH]ccn2nnnc12)N(C)C(C1(F)CC2(CCC2)C1)=O C(=O)(C1=CCCN(C(c2cnc(N(C)C)o2)=O)C1)Nc1cn(CCC#C)nc1 C1(NC(CCCC)=O)CCCC(NC(c2cocc2Br)=O)CC1 n1(CC)cnc2nc(=NCC=CCl)[nH]c(NCC3(CO)CCC3)c12 N1(C(CC(OCC)OCC)=O)CC2CCN(C(C3(F)CCCC=C3F)=O)C2C1 CC#CCCC(=O)NCCCN(C(c1cnc(CC(C)C)s1)=O)C1CC1 C(CCC(F)(F)F)ONC(CN(C(CC)C(=O)Nc1cccc(F)c1)C1CC1)=O C12(C(=O)NCCC(C)(C)NC(c3cc(Cl)ccn3)=O)CCCCC1CS(=O)(=O)C2 N#CC1CC2(CC(OC(=O)C=Cc3csc(C(F)(F)F)c3)C2)C1 C1(C(N(CC(C)NC(=O)CC2COCCOC2)C)=O)CCCCCN1C c1(OC)ccc(C(=O)NC2CCN(C(=O)C(C3CC3)OC)C2C2CC2)cc1F c1(C(N(CCCNC(c2cnncc2O)=O)CC)=O)ccc2c(c1)CCC(O)C2 C(C(F)(F)C(=O)NCCCC(=O)NC(c1nncs1)C)OC CC1CC(NC(c2cc3occc3[nH]2)=O)CCN1C(=O)CC1CCC2CC2C1 N1(C(CSN2CCN(C)CC2)=O)CC(C(COC(C=C)=O)C)CCC1=O C1(C(C)NC(COCC)=O)CCN(C(=O)CSc2nncn2C)C1 CC(N=c1[nH]c(=NCc2nnc(O)o2)[nH]c2c1COC2)c1ncc(Br)cn1 CCC(C)C(CNC(=O)C(Cc1cnc[nH]1)NC(=O)Cn1ccnn1)OC CC1=C(CCCN(C(=O)CC(C)C(C)C)C(=O)Cc2nn[nH]n2)COCC1 Cc1cc(C(=O)NCC(C)(C2CCC2)NC(=O)C2=CCOC2)c2n[nH]cc2c1 N1(C(c2c(C)cn(C)c2)=O)CCC2(CC(C(=O)N3CC(O)CCO3)C2)C1 N1(C(C(C)(C)n2cccn2)=O)CC2CCCC(NC(c3ccc(F)s3)=O)C2C1 N1(c2nc(C)cc(CC)n2)CC(C)CN(C(c2n[nH]cc2Cl)=O)CC1C C1(CNC(C(C)CN(C(=O)C=Cc2cccnc2)C)=O)CCC2(CC2)CO1 C1(OCC)CN(C(=O)C(c2ccc(F)cc2)(F)F)CC1CNC(=O)C(F)=C(C)C N(C1CCCn2ncnc21)C(C(CCC)NC(c1ccncc1Cl)=O)=O c1(C(=O)NC(CCC)CCO)nccc(C)c1F C1(C(=O)NC2(C)CCCC2(F)F)CC2CC1CN(C(=O)CCc1ccncn1)C2 c1(C(=O)NC2C(C(=O)NC(c3nnnn3C)C)CC2)nccc2cc[nH]c12 N1(C(c2nc(C)oc2)=O)CCC2(C1)CN(C(c1csc(C)c1C)=O)CCO2 CN1C(=O)CCCC1C(=O)NC1CCCCN(C(c2cnn(CCF)c2)=O)C1 N1(C(CC(OCC)OCC)=O)CCOCC1CNC(C1CC(C)C1)=O N1(Cc2c(C)nc(C)o2)CCCC1C1CCCCN1C(C1(F)CCCC1)=O C(=O)(CCCCOC)NCCN(CCC)C(c1cc(C2CCCO2)n(C)n1)=O Cc1ccc(S(=O)(=O)C2(C(N3CCN(Cc4cscn4)CC3)=O)CCCC2)cc1 c1(C(=O)NC2CN(C(=O)Cc3cc[nH]n3)CC2C(F)(F)F)occ2c1CCCC2 C(=O)(C(C)(O)C(F)(F)F)NCC(C(C)(C)C)OC.N12CCCC1C2=O c1(C(N2CCC(O)(CN(C(Cc3c(C)noc3)=O)C)C2)=O)coc2c1COC2 Nc1ccc(C(=O)NCC2CCN2C(C2CCCCCCC2)=O)cc1N N1(C(Cc2n(C)ncc2)=O)CCOC2(CCCN(C(c3ccc(Cl)nn3)=O)C2)C1 C(=O)(C1CCCc2cc(O)ccc21)NCc1c(F)ccc(OC)c1 CC(Cc1ccnn1C)C(=O)N1CCC(CNC(C2(c3cccnc3)CC2)=O)C1 N1(C(CC(CC)(C)C)=O)Cc2n[nH]cc2C1C(=O)NC1CCCC2(C1)N=N2 N1(C(CN(C(C(C)N(C(C)=O)CCO)=O)C(C)C)=O)CCOCC1 C1(NC(CCOCCOCC)=O)CCCC(NC(c2n[nH]cc2C2CC2)=O)C1 CC1(C(=O)NCC(O)CCNC(c2cncc(N)c2)=O)CCCNS1(=O)=O c1(OC)ccc(F)c(C(=O)NC(CC=C)CNC(C2CCN(C3CC3)CC2)=O)c1 CCCC(C#N)C(=O)NC1CCC(NC(=O)C(n2nnnc2C(C)(C)C)C)CC1 N1(C(CCC=CCC=C)=O)C2CCC1CC(CCNC(=O)C(O)C(F)(F)F)C2 c1(CNC(C(C)c2cc[nH]n2)=O)ccc(CCNC(C2(N(C)C)CC2)=O)cc1 c1(N(C)C(C2COCC2NC(C2(Cl)CCC2)=O)=O)cccc(C#N)c1 c1(SC)nc(Br)c(NC(c2nc(NCc3[nH]cnc3C)cn2C)=O)n2ccnc12 c1(-c2ccc(SC)cc2)cnc(NC(c2cn(C(C)(C)C)nn2)=O)c(O)c1 N1(C(C2(N(C)C)CCC2)=O)CCCC(CNC(=O)Cc2nn(C)cc2Br)C1 CC1(C)CCC(CC(=O)NCC2CC(NC(=O)C(C)(C)CCF)C2)CC1 Cn1c(C(=O)NC2CC(NC(C3(c4cc[nH]n4)CC3)=O)C23CCC3)cccc1=O C1(N(C(C=CSC)=O)CC2CCCO2)CCN(C(C2NC(=O)C3CC23)=O)CC1 Cc1ccc2oc(C(=O)NCC3CC(NC(=O)CSc4n[nH]c(O)n4)C3)cc2n1 C1(C(=O)NCc2ncc(CC)o2)CCC2(CC2)N1C(=O)Cc1ccns1 c1(NC(C2CCCN2C(c2csc([N+](=O)[O-])c2)=O)C)nccc(S(C)(=O)=O)n1 c12cc(F)ccc1C(=O)N2.c1(C2C(C(=O)OC)C2)nc(C2CC2)cs1 C1(c2ccc(C)cc2)CCN(CC2CCS(=O)(=O)N2C)CCO1 c1(N(CCCNC(C2(OC)CCSC2)=O)C(C)C)nc2cccc(C)c2s1 c1(SC)ccc(C(=O)N(CC(=O)N(C)C2CC2)CC2CCSC2)o1 C1(NC(c2ccc(C(=O)OC)s2)=O)C(C)(C)C(NC(=O)C(C)C(C)(F)F)C1(C)C C=CCC(C)(C)CC(=O)NC1CCCC(NC(=O)C(CO)N(C)C)C1 CC1CCCC(CC(=O)NC(C)(C)CN(C)C(c2cc(O)ncn2)=O)C1 C(=O)(CC(C)C(F)(F)F)NC1C(C(=O)Nc2c(C)cccc2)CCC1 CC1CCC(C(=O)NCC=CCNC(=O)CCC2CCCCC2)C1 CC(C)C(F)C(=O)N1CCC(C)(NC(c2ccc(Cl)cc2)=O)C1 C1(CNC(CCOCCC)=O)CC2CN(C(=O)C(N3CCCCC3=O)C)CC12 C(=O)(C(O)CC(F)(F)F)NC(CNC(c1ccc(CC)cc1O)=O)(C)C1CC1 c1(OC)cnc(Cl)cc1C(=O)NCCCC(C)NC(c1ccc(Cl)cn1)=O CCCS(=O)(=O)CC(=O)N1CC2(CC)CC1(CNC(=O)CC(C)C(C)C)C2 C12(NC(C(=Cc3cccs3)C)=O)CCC1CN(C(C1(C)CCC(=O)N1)=O)C2 Cc1nc(C(=O)NCC(C)N(C(=O)C(F)(F)C2(O)CCCC2)C)c(C)o1 N1(C(C2CCC(C)N(C(=O)Cc3cn[nH]c3)C2)=O)CCC(C2CCCC2)C1 Cn1nc(C(=O)NC2CC(F)(CNC(C3(O)COC3)=O)C2)c2c1CCC(F)(F)C2 N1(C(c2ccc(COC)o2)=O)CCN(C(C2CC3C=CC2O3)=O)C(C)C1 N1(C(C(c2ccco2)NC(C(C)=CCC)=O)=O)CCCC1CN(C)C c1(SCC(=O)N(CC(C)NC(c2cnco2)=O)C)ccccc1 CC1=C(C(=O)NCC2CCN(C(=O)CCCCC(C)C)C23CC3)C(C)(C)CCC1 C1(C(=O)NCC2C(NC(C(C(C)C)N(C)C)=O)CCCC2)CCCCC12CCC2 C1(C(=O)NCc2cc(C)on2)CCC(NC(=O)C(F)C(C)C)CC1 C1(O)(C(CNC(C2N(CC)CC2)=O)C)CCN(C(=O)CCNC(N)=O)C1 C#CCC(CC(F)F)NC(C1COCC1NC(=O)C(C)OCC1CC1)=O C(=O)(C(C)S(C)(=O)=O)NC(CSC)CCn1cc(-c2[nH]c(=NC)sc2)nn1 Nc1cncnc1C(N1CCCCC1C(=O)NCCC1CCSC1)=O C#Cc1ccc(F)cc1C(=O)NC1CN(C(=O)CC2CC(=O)C2)C(C)(C)C1 c1(C(N2CCC(C)SCC2)=O)ccc2c(n1)CN(C(=O)CCCN=[N+]=[N-])CC2 N1(C(C(SC)SC)=O)CC(C)CN(C(C2CCCC23CCC3)=O)C(C)C1 C12(CNC(C(c3ccccc3)OCC)=O)CC(NC(C3CC3F)=O)(C1)C2 c1(CC)c(NC2CCCN(C(=O)CC(C)c3cnn(C)c3)CC2)ncnc1Cl CC1CC(C(=O)NCCCCC(C)NC(c2cnccn2)=O)CCC1=O Cc1cccc2[nH]c(C(=O)NCC3CCN3C(=O)CCCC(=O)NC(C)C)cc12 N1(C(c2ncn(C(C)C)n2)=O)CCC(O)(C2CCN(C(C3(CF)CC3)=O)CC2)C1 Cc1cc2nc(Cl)[nH]c(=NC(C)CC(C)NC(=O)CC34CNC(=O)C(C3)C4)c2s1 c1(OCC(N2CC(CC=C)(NC(C3CCN(C)C3=O)=O)C2)=O)ccccc1CC N1(C(COc2ccc(CSC)cc2)=O)CC(O)(C(=O)O)CC1(C)C c1(COC(C(n2c(C)cc(C(F)(F)F)n2)C)=O)ccc(Cl)cc1C(F)(F)F N1(C(C=CC(CC)C)=O)CCC2(CC1)CN(C(c1nc(Cl)oc1C)=O)C2C(C)C C1(NC(C2(N(C)C)CC2)=O)CC2CCC1CC2NC(c1ccnc2[nH]ncc12)=O C1(C(C(=O)NCc2cccs2)CC(=O)N(CC(=O)OC)C)CC2C=CC1CC2 N1(C(c2c(CCC)nco2)=O)CCC(NC(=O)C(C)CCOC)CC1C c1(C(=O)NCC2N(C(C3C(C)OC(C)C3C)=O)CCC2)ccc([N+](=O)[O-])cc1F c1(C(=O)NC(C(C)(C)C)CNC(C2(C(C)(C)O)CC2)=O)cn2c(n1)CCC2 c1(-n2cc(CN(C(C3CCN(C(C)=O)CC3)=O)O)nn2)cc(C)ccn1 c1(CN2CC(CC(=O)Nc3ccnc(C4CC4)c3)OCC2)ccc2sccc2c1 C(CC(=O)NC1(CF)CCCC1)(C(F)F)CNC(CN1CCC(OC)C1)=O N1(C(c2ccn(C)c2)=O)CC2CC(NC(=O)CC3CC3C(F)(F)F)C(C2)C1 c1(NC(C2CC(NC(CC(=O)OCC)=O)C2)=O)ncc(C2CC2)cc1F C1(C)(CCC(=O)OC)CCCN1CC(=O)NC(c1ccccc1N)(C)C c1(CC(N2CCN(C(CC(CCC)O)=O)C(C)CC2)=O)ccc2c(c1)OCCO2 C(c1cccc(Br)c1)=CC(=O)NCC(CC=C)NC(c1cnc(O)n1C)=O n1(C(C(C(=O)N(C2CCOC2)CC)C(C(C)C)OC)CC)ncc2ccccc12 N1(C(C2C(C)C2C)=O)CC(CNC(C2(N3CCOCC3)CC2)=O)CC1(C)C c1(CC)oc(C(=O)NCC2CC2NC(c2cnc(-c3cnn(C)c3)s2)=O)cc1C C1(N(C(C2CCC(COC)O2)=O)C)CCN(C(=O)C#CC(C)C)CC1C C12(CNC(COCC)=O)CCCC1CN(C(C1(F)C3CCCCC13)=O)C2 c1(C(N2CCCN(C)C(=O)C2)=O)cc2cc(Br)cnc2o1 N1(C(c2cc(CC)nnc2C)=O)CC2CCC(NC(=O)C=CC(C)C)(C2)C1 c1(CC(=O)NCC2(O)CN(C(C3(OCC)CCOC3)=O)C2)cn2c(C)csc2n1 c1(C(=O)NC2(CO)CCN(C(C=C3CCC(C)C3)=O)C2)[nH]cc2c1CCC2 C1(CNC(C(C2CC2)OCC)=O)CCC2CN(C(C3(SC(C)C)CC3)=O)CC12 C(=O)(CC(C)CC(=O)NC(C1CCN(C(c2ccc(Cl)c(F)c2)=O)C1)(C)C)OC O=S(=O)(NC(CO)C1CC1)N1CCN(N2CCN3C(=CN=C2C(F)F)C3)CC1 C(=O)(CCCCC(F)F)NCC(CCOC)NC(=O)C(C1CC(F)(F)C1)OC C1(C(C)C)CN(C(=O)CC(C)CF)CCN1C(c1cn(CCO)nn1)=O c1(C(CC)O)nc(-c2csc(Sc3ccc(C)cc3)n2)n(Cc2ccccn2)n1 c1(C(=O)OCC(=O)NC(C(=O)OCC)C2(C)CC2)ncc(OC(C)(C)C)cn1 C(=O)(C(c1ccco1)NC(=O)CCn1cccc1)N(CCCO)CC CC(CC(=O)N(C)CCOCCC(=O)NC(C)(C)CC1CCC1)C1CC1 C1(NC(C(CC=CC)C)=O)(CNC(=O)CCCCC2CC2)CCCCCC1 N1(C(C(C#C)(C)C)=O)Cc2ccc(C(C)NC(c3cnn(C)c3)=O)cc2C1 c1(C(=O)NCC(C)(C2CCC2)NC(C2N(C(C)=O)CCC2)=O)nccc(Cl)c1C C1(C(N2CC3C(CNC(CCC=CC)=O)C3C2)=O)CCc2nn(C)cc2C1 CC(C)CS(=O)(=O)CC(=O)N1CCCC(CN(C(=O)C2=CCCOC2)C)C1 C1(CC)CCc2nc(CNC(N3CCCCC3c3ocnc3C(=O)O)=O)sc2C1 N1(C(C(CCC)CC)=O)CCC(C2CCN(C(c3ncc(N)nc3C)=O)C2)CC1 c1(C(=O)NCC(Cn2cc(C(C)(O)C(=O)O)nn2)OC)occc1C(C)C Cc1ccc(NCc2ccc(OCC#N)cc2)c2c1CCC2 C12(CNC(=O)C3=CCCCO3)CN(C(=O)C3=CCCS3)CC1CS(=O)(=O)C2 Cn1nccc1C=CC(N1CCC2C(NC(=O)CCc3ccccc3)C12)=O c1(CC)[nH]nc(Cl)c1C(c1nnnn1C1CCC1)NCc1ncco1 C(=O)(CCCCCNC(=O)CC1CCC(C)(C)C1)NC(C)C(=O)N(C)C C(=O)(C#CC1CC(F)(F)C1)NCC1CCCN(C(C=C2CCC(C)CC2)=O)CC1 c1(NC(c2ncc(-c3ccc(OC)cc3)o2)=O)cc2c(cc1Br)OC(F)(F)O2 Cc1cc(C)c(C(=O)NCC(C2CC2)N(C)C(C2CCCC(O)C2)=O)cc1N CCC(CC)(CC)C(=O)NCC1(NC(C2CC(C#N)(OC)C2)=O)CCCCC1C CCCCCC(O)C(=O)N1CCN(C(=O)CC(F)F)CC1CC1CC1 C1(CC)(CNC(=O)C(C2(C)CC2)NC(C2CN(C3CCC3)C2)=O)CCOCC1 N1(C(CC2C(C)=NOC2=O)=O)CC2(C1)C(NC(c1cc(C)ns1)=O)CCS2(=O)=O c1(OCC)nc(C(N2CC(C(C)NC(=O)CN(C(=O)COC)C)C2)=O)co1 C=CC(C)(CCOC)C(=O)NCCN(C(c1cscc1C(N)=O)=O)CC c1(C(=O)NC2C(C)CCN(c3c(F)cnc(C)n3)C2)ccc2nnn(O)c2c1 CCCCC(=O)NC(C1(O)CN(C(=O)CCSC2CCCC2)C1)C C1(CNC(c2cc(C)sc2)=O)CC2(CO1)CN(C(=O)C(C)(C)c1ccncc1)C2 Cc1ccccc1C1CC1C(=O)N(CC(C)O)CCNC(=O)CCc1cc[nH]n1 Cc1cc2c[nH]nc2c(C(=O)NCC(CO)NC(C2CC(F)C(=O)N2)=O)c1N c1(C(N2C(C)C(NC(=O)CC3CCC(=O)N3)CCC2)=O)cc2nc(Cl)ccc2s1 CON1CCC(CC(=O)NCC(C)(C)CN(C)C(C23CC4CC2C3C4O)=O)CC1 C1(NC(C2=NOC(CNC(=O)CC(=O)NCC3CC3)C2)=O)CC2OC(=O)CC12 c1(C(=O)NCC2C(C)CN(C(=O)CNC=O)C2)ncsc1S(N)(=O)=O CC(F)(F)C(C)(C)C(=O)N1CC2(COC(CNC(=O)Cc3ccc(Cl)nc3)C2)C1 c1(C(=O)NC(CC)(CNC(c2nc(Cl)sc2C)=O)CC)ccc2ncncc2c1 C1(CCC)CCC(C(=O)Nc2nc(N3CCCC3)ns2)CC1 c1(CN(c2nccc(Cc3ccc(F)cc3)n2)C)ccc2occc2c1 c1(C(N2CCC(CC(=O)Nc3cc(C)nc(C)n3)C2)=O)cc2ccc(Cl)nc2[nH]1 CC(C(=O)N1CCC(CNC(c2cccc(C(C)(C)C)c2)=O)C1)C(C)(F)F N1(C(C2CN(C(C(C)SC)=O)CC23CC3)=O)C2C=CCC1CCC2 c1(C(=O)NCCC(C)NC(C23CCCCC2C3Br)=O)cccc(F)c1F N1(C(C=CC=CC)=O)CCN(C(c2ccc(C(C)(F)F)cn2)=O)C(C)CC1C CC(C)(C)CCC(=O)N1C2CCC1(CNC(=O)Cc1csc(C(F)(F)F)n1)CC2 C1(CNC(C2(C#C)CC2)=O)C2CN(C(c3cn(-c4ccccc4)cn3)=O)CC12 c1(NS(=O)(=O)CC2CC23CCCCC3)ccc2ncc(Cl)n2c1 c1(OCC(CN2CC(C)(CNC(c3cc(C4CC4)on3)=O)C2)O)cc(Cl)cc(Cl)c1 C1(CNC(c2ccc(C(C)C)o2)=O)CCN(C(C2CC2C2CCCO2)=O)CC1O C(=O)(CCCC(C)(C)C)NC1CCC(CNC(c2c(CSCC)cccn2)=O)C1 c1(C(C(=O)NC(C)CC2CN(C(c3cnco3)=O)C2)OC)cnn(C)c1 N1(C(c2ccn(CCOC)n2)=O)CC2OCC(C(=O)NCCCOC(C)=O)C2C1 c1(C(N2CCC(NC(C3CC(O)(CC#C)C3)=O)C2)=O)ccc(S(C)(=O)=O)[nH]1 c1(NCc2ccc(NCc3c(C#N)cccc3)nc2)cc([N+](=O)[O-])c(F)cc1Cl C1(OC)CCN(CC(N2CCCC2C(=O)NC2C=CCC2)=O)C1 c1(C(=O)NC2CCCC(NC(C(C)SCC)=O)C2)cc2c(=O)[nH]c(C)cn2n1 c1(C(C(N2C(CNC(c3ncn(CC)n3)=O)CC2)=O)O)ccc(Cl)cc1F c1(OC)ncc(C(=O)N(CCC(=O)NC2CCOC2)C(C)C)cn1 C(=O)(C(CN=[N+]=[N-])NC(=O)CC(C)O)N1CCN(C(=O)NC)CC1 c1(NC2C(C)CCN(C(c3cccc(=S)n3O)=O)C2)ncc2c(n1)COC2 c1(SCCC(N2CCC(NC(CC(C)SC)=O)C2C)=O)ccccc1[N+](=O)[O-] N1(C(C2C(=C)C2)=O)CC(F)(F)CC1CNC(=O)C(C1CCOC1)OC C1(NC(C(=O)N(C)C)=O)CCC2(CCN(C(=O)C(C)(C)S(C)(=O)=O)CC2)C1 CN1C(=O)CCC1C(N1CCSCC1CCNC(=O)Cc1ccco1)=O C(CC1CC1)(C(=O)NCC(C)C(=O)NCCC(=O)N(C)C)OC c1(C(N2CC(C(C)NC(c3cc(C)no3)=O)C2)=O)cccc2ncccc12 CCC(C)CCC(=O)N(C(CC(F)F)C(=O)NC1(CCCF)CC1)C N1(C(C(CC=CC)C)=O)CCOCC(NC(c2ccc(C3(CC)CC3)cc2)=O)C1 O=C(CCCc1ncco1)NC1CC(NC(C2CCC2)=O)C1 c1(CNC(NC(COC)C)=NCC(C)NC(C)=O)nn(C)c2c1COCC2 CN1CCC(C(=O)NC(Cn2cccn2)CO)(NC(=O)C=C2CCCCC2)C1 c1(CC(=O)N(CC(CC)NC(=O)CC2CSCCS2)C)cnc2cccnn12 N1(C(c2cc(CCC)on2)=O)CC(C)(C(=O)NOC2CCOC2)CC1(C)C N1(C(c2nc(COC)oc2)=O)CC(NC(=O)COC2CCCCC2)CC(O)C1 C1(OC)CN(C)C(C)(C(=O)NCC(CC(C)C)NC(=O)CCNC(C)=O)C1 c1(C(=O)NCC2(O)CC(NC(=O)C(Cl)=CCl)C2)cc(O)nc(O)n1 CC1CCN(C(C2COC(=O)N2C)=O)C(C(=O)N(C2CCCC(O)C2)C)C1 CCC(CC(=O)NC(C1CC1C(N1CCCC(C(=O)NC)C1)=O)C)CC(C)C C12(C(=O)NCCOCCNC(C3(C)CCNC3=O)=O)CCC(C)(C1)OC2 C1(CC)CCCCC1C(=O)NCC1CCN1C(c1conc1C1(C)COC1)=O N1(C(c2c(C)cc[nH]2)=O)CC2CC1C2NC(c1cnns1)=O C1(C(N(CC(CC)O)C)=O)CN(C(c2nccn2C)=O)CC1(F)F c1(C(=O)NC2CN(C(=O)COCc3ccccc3)C2)c(Br)cc(Br)c(O)c1Br c1(C(c2nnnn2C(C)C)NC2CC(OCC)C23CCC3)cc(Cl)c(C)cc1Br c1(CC)nnc2n1CCCC2C(=O)N(CCCNC(=O)C(C)S(C)(=O)=O)CC c1(NC(c2c(NC(C3C(C(=O)OC)C3)=O)cnn2C)=O)cccc2c1C(=O)CC2 Cc1cccc2cc(C(=O)NCC3CCCC(NC(C4CC(O)C4)=O)C3)cnc12 N1(C(c2c(C#C)cnn2C)=O)CC2CC(NC(C3CC=C(C)CC3)=O)C(C2)C1 c1(C(=O)NC(c2ccccc2)C(=O)NC2CC(CC)C2)ccc2[nH]nc(Cl)c2c1 C1(NC(CN(CCC)C)=O)CCC(N(C)C(c2cc(C3CC3)ccn2)=O)CC1 C12(CNC(c3cnccn3)=O)CCC(CN(C(c3cc(F)c[nH]3)=O)C1)C2 c1(OCC(C)C)ccc(CCNC(=O)N(CCS(C)(=O)=O)C)cc1 C(=O)(CCCCC(=O)N1CCCC1C1(C(=O)Nn2cccn2)CC1)OC N1(C(C(C(C)C)n2ccnc2)=O)CC(NC(c2ncn(C(C)C)n2)=O)CC(F)C1 c1(CNC(CN(C2CC2)CC)=O)ocnc1C(=O)NCCCC(OC)OC C1(CNC(CCNC(CC=C)=O)=O)CCCN1C(C1CC(C)(F)C1)=O N1(C(CCc2c(C)cccc2)=O)CCCN(C(=O)CCc2ccsc2)CC1 c1(OC)c(F)ccc(F)c1C(=O)N(CCCOCCNC(C1CCCC1O)=O)C c1(C(=O)NC2CN(C(=O)CC3CCC3)C3CC23)cc2nccn2c(O)n1 C1(O)(C(=O)NCC2(CC(=O)NC(CC)C(C)O)CC2)CCSCC1 N1(C(COCCC#C)=O)CCC2(C1)CN(C(c1cnc(S)nc1)=O)CC(C)O2 Cc1nn[nH]c1C(=O)NCc1cn(CC2CCCN2C(C2CC2CF)=O)nn1 N1(C(C(C(C)C)n2cccc2)=O)CCN(C(C2CNC(=O)N2C)=O)C2(CCC2)C1 C1(CN(C(C2C(COC)C2)=O)C)CCC(CNC(=O)C=CC(F)(F)F)CC1 c1(C(=O)OC)ccc(-c2cn(C3CC(C(c4cccc(Cl)c4)=O)C3)nn2)cc1C C12(NC(C=C(CCC)C)=O)CCCC1CN(C(c1ccn3cncc3c1)=O)C2 CC(CSC(F)(F)F)C(=O)N(CC(O)CNC(c1ccccc1)=O)C C1(CC(N2CC(CCC)OCC2)=O)C2CCCC2N1C(C1CC12CCOCC2)=O CCC(F)(F)CC(=O)NCC12CC1CN(C(=O)CC1CCCC1)C2 C=C(C)CC(C(=O)N(CC(C)NC(c1cc(O)nc(O)c1)=O)C)NC(C)=O C1(NC(c2cc(C)sn2)=O)CCCN(C(c2cccc(OC(F)F)c2)=O)C1 N1(C(c2c(OC)cc(C)cn2)=O)C2CCC1CN(C(c1coc(C(C)C)n1)=O)C2 C(c1ccncc1)=C(C)C(=O)N(CCC(C)NC(C1CC(NS(C)(=O)=O)C1)=O)C N1(C(c2c(C)[nH]nc2C(C)C)=O)CC2CC(NC(=O)C(F)CC3CCC3)C1C2 N1(c2ccnc(OC)n2)CCC2CN(C(=O)CC3CCCCO3)CC12 c1(C(N2C3CN(C(C4CC(C)(C)C4)=O)CC32)=O)ccc(I)c(F)c1 C1(N(C2CCCCC2)C(COC(C(C=CC)O)=O)=O)CCOCC1C C1(CC(=O)NC(C2N(C(c3c(OC)n[nH]c3)=O)CCC2)C)CCC(C)CO1 C1(C(=O)NCCNS(CCC)(=O)=O)CC1C1CN(C(=O)OC(C)(C)C)C1 N1(C(Cn2c(C)ccn2)=O)CC2CC2(NC(C2COCC2(C)C)=O)C1 N1(CC(C)NC(C2CCCCC2C)=O)CCCC(O)C1c1ccccc1 c1(CN2CCC(C(=O)Nc3ccccc3-n3cncn3)CC2)cccc(O)c1F Cc1c(C(=O)NC(C)CC(C)NC(c2cnn(C)c2Br)=O)ccn1C C12(C(N(C(C)C3CC3)C)=O)CCC(CC1)N(C(C1CNC(=O)C1)=O)C2 c1(C(=O)NCCC2CN(C(C3C(CC)CCCC3)=O)C2)ccn2cnnc2c1 c1(C2CCC(NC(=O)NCC3N(C(=O)OCC)CCC3)C2)cccc(F)c1 C1(NC(c2cc(SC)oc2)=O)CCOCC1NC(=O)CCOC(C)C c1(C(N2CCC(NC(c3cc(C)[nH]n3)=O)C2)=O)ccccc1N(S(C)(=O)=O)C Cc1cc(-c2nc(CCO)nn2C2CCC(C)(C)C2)n2nccc2n1 c1(C(=O)NCC2CC(NC(c3cnn(CC)n3)=O)C2)cccc2c1ccn2C c1(C(=O)NC(C23CC(CO2)C3)C)cc(CNC(C2CN3CCC2C3)=O)nn1C C#CC1(C(=O)Nn2cnnc2)CCN(C(C2CC(O)C(F)C2)=O)CC1 Cc1ncc(NC(C2C=CC(NC(c3cc(Br)cnc3C)=O)C2)=O)cc1F c1(CNC(CN(C(COC)=O)C)=O)occc1C(=O)NC(C)C(C)CO C1(NC(CC2C(C)(C)C2)=O)CN(C(C2CC23CCOC3)=O)CCC12CCOCC2 CC(C)C(F)(CNC(c1cc[nH]c1)=O)C(=O)NCC1CC2(CCC2O)C1 c1(C(=O)NCCC(C)NC(c2ccn(C3CCC3)n2)=O)coc2c(Cl)cccc12 C(=O)(C(C)(C(C)C)OC)OC(c1ccc(CC)cc1Br)C C1(NC(C2(C)CCCN(C(C3CC4(CC4)CO3)=O)C2)=O)CC2(C1)CC21CCC1 c1(OC)ccc(O)c(C(=O)NCC2CCN2C(c2oncc2C)=O)c1 c1(NC2C(C)(C)CN(C(C3(Br)CC3)=O)C2)ncc(Br)cc1C#N N1(C(Cc2cccc(COC)c2)=O)CCC2CN(C(=O)C3=NOCC3)CC2CC1 c1(C(=O)NC(C2(O)CN(C(=O)Cn3ncnn3)C2)C)ccc(Br)c(F)c1 C(CCCC(=O)NC1CC(CC(=O)NCC2(C)CCN(C(C)=O)C2)C1)SC c1(C(N2CC(OC)C(NC(=O)C=CCO)C2)=O)ccc(Cl)cc1OC(C)C O=C1CCCC(C(N2CCC(F)(CNC(c3cc(C(F)F)[nH]n3)=O)CC2)=O)CC1 C(=O)(C1=C(Cl)CCOC1)N1CC(C(C)C)N(C(=O)CC2(O)CCCCC2)CC1 C=C(Cl)CCC(=O)N1CCOCC1CN(C(=O)C(n1ccc(Br)n1)C)C c1(OCC)ccccc1C(=O)NC1CC1NC(=O)C(c1cccc(Cl)c1)C C123CCC(CC1)(C2)Cn1cc3nn1.Cc1nn[nH]c1C1CN(C(=O)CC(C)O)C1 C=CCC(C)(C)C(=O)N1CC(O)(CNC(C2(C(F)F)CCCC2)=O)C1 C12(CNC(=O)CCN3CCOCC3)CCCCC1N(C(c1csnc1Cl)=O)CC2 Nc1ccc(-c2nc(CCOC(F)(F)F)n(CC3CCCCN3)n2)cc1 C1(N(C(CC=CC=C)=O)CC)CCN(C(c2cc(C(C)(C)C)ccn2)=O)CC1 c1(C(=O)NCCCN(C(=O)C(C)(C)c2cncnc2)C)cn2cc[nH]c(=O)c2n1 C1(OC)(CNC(c2ccnn2C(C)(C)C)=O)CC(OC)C1.C12CC(C1)N(C)C2=O N1(C(CCSC)=O)CCN(C(c2cc(C(N)=O)n(C)n2)=O)C(C2CC2)C1 c1(OC)ccc(Cl)c(C(=O)Nc2nc(CC(N3CCC(NC(C)=O)C3)=O)cs2)c1 CC1CN(C(CCCC2CC2)C(=O)NC(C2CC2)C2CC2)CC2(CCOC2)O1 Cc1ccc(C)c(OCC(=O)NC2CC(NC(C3CC(=O)OC3(C)C)=O)C2)c1 Cc1ccc(F)c(C(=O)NCc2ocnc2C(=O)NCc2nc(C)no2)c1 c1(OC)ccc(Br)c(CN2CCCC2C(=O)Nc2ccc(C3CC3)nc2)n1 c1(NC(c2cc(OCC)ncc2-c2ccc(C)nc2F)=O)c(F)cc(F)cc1Br c1(C(=O)NC2CC(CCNC(C3(C)CC3(Cl)Cl)=O)C2)c(C2CC2)cccc1F C1(CNC(C(C)N(C(=O)C(F)F)CCC)=O)CC(CC)=NO1 C(C1CCc2nccn21)NC(C1(CC)CCN(C(=O)C=C2CCC(C)CC2)C1)=O N1(C(CCC(C)(C)NC(c2c(C)ccnc2C)=O)=O)CC(C)(C)C2COCC12 c1(CNC(C(N2CCOCC2)C)=O)cc(Cl)c(Cl)cc1Cl C1(OC)CC2CC(C1)N(c1cc(Nc3ccc(CNC(=O)OC)cc3)ncn1)C2 C(CC(F)Cn1cc(C(C)O)nn1)NC(CNC(CCC)=O)=O CCC(CCCC(=O)N1CC(NC(=O)OC)C1)NC(=O)Cc1ccon1 C1(NC(C(COC)(F)F)=O)CN(C(=O)C(C)n2ccnn2)CC2CCCC12 C1(CCO)(NC(C2C(=C)CC2)=O)CN(C(=O)CC(C)c2ccccc2)C1 Cc1cc(F)ccc1C(=O)NCCCN(C(=O)C(F)C(C)C)C(C)C c1(CC2(C(=O)NCC(C(=O)OC(C)C)C)CC2)ccc(Br)cc1 C(=O)(CC(C(F)F)NC(c1ncncc1Cl)=O)NCc1ccnc(OC)n1 C#Cc1ccc(C(N2CCCC2C2(NC(=O)CSC3CC3)CC2)=O)c(F)c1 c1(NC(C2N(Cc3cccc(OC)c3O)CC2)=O)cc(F)c(I)cc1C C(=O)(CC(C)(C)C(F)F)N1CCC(NC(Cc2c(C)ccs2)=O)(CF)C1 c1(C(=O)NC(CCCNC(c2ccc(-c3nc(C)sc3)s2)=O)C)ccccc1F n1(CC(=O)NCC(C)(C)CNC(C2CC3CC2C2CC32)=O)ncc(O)nc1=O c1(C(=O)Nc2ccc(F)nc2)cc2cccc(-c3cnc(N4CCC4)nc3)c2s1 N1(C(C(n2cc(Cl)cn2)C)=O)CCC2CCN(C(C3CC4(CCC4O)C3)=O)C2C1 C=CCC(C(=O)N(CCCOC(C)C)C)NC(C1C(C)(C)C1(F)F)=O C1(NC(C(C)CCO)=O)CC2CN(C(=O)Cc3cc[nH]n3)CC12 N1(C(COC(CC)(C)C)=O)CC(O)CC1C(=O)NC(C)Cc1nc[nH]n1 c1(CC(N2C(CCNC(C3C(CC)CCO3)=O)CCCC2)=O)c(O)ncnc1O C1(OC)CC(CNC(=O)CSC2CC2)(NC(C)=O)C1 N1(C(CCOC)=O)CC2CC(C1)C2NC(c1cc(C)[nH]c1C)=O n1(CC)ncc(C)c1C(N1CCC(Oc2ccncc2)C1)C(=O)NCCSC n1(CCC(=O)NC(CCNC(c2cc(C)no2)=O)C)cc([N+](=O)[O-])nc1C C1(C(=O)NCC(=C)CCNC(=O)C(C)(C)N(C)C)(CSC)CCOCC1 c1(NC(C2CCC(C(=O)OCC)C2)=O)ccc2c(c1)nnn2C CC(C(=O)NCC1CC(NC(c2cn3ccnc3s2)=O)CC1O)S(C)(=O)=O CC1CCc2c(C(=O)NCC(C)N(C)CC34CCCN3CCC4)csc2C1 C1(CC(=O)NC)CN(C(=O)Cc2ccccc2C)CCN1C(=O)C(O)C(F)F C1(C(=O)NCC2N(C)CCN(C(CN(C(C(C)C)=O)C)=O)C2)CC(C(C)(C)C)=NO1 Cc1nn(C)c(Cl)c1C(=O)NCCC1COCCN1C(=O)CC1CCCC(=O)N1 Cc1nc2cc(C(=O)NC3CN(C(c4cc5nccn5c(O)n4)=O)C3)cnc2[nH]1 N1(C(c2c(Cl)cc(C)nc2)=O)CCC2CN(C(c3cc(C4(C)CC4)n[nH]3)=O)C2C1 N#CC1(C(=O)NCCc2n[nH]cc2C(=O)NCCCN=[N+]=[N-])CC=CC1 c1(C(=O)NCC2COCCN(C(c3ccc(C)[nH]3)=O)C2)c(C)nc2ccccn12 c1(C(C)=O)ccc(NC(C2CCN(C(C3CC3(C)C)=O)C2)=O)c(F)c1 c1(C(=O)NC(C(CO)NC(c2c(C)nn[nH]2)=O)C)cnn2ccc(Cl)c(F)c12 N1(C(C2CN(C(CCN(CC)CC)=O)CC2(C)C)=O)CC2CN(C)CC2(C)C1 N1(C(CC(CC)NC(CC=CC)=O)=O)CCc2c(cnn2C)C1 N1(C(Cc2ccc(C)s2)=O)CCOCc2cc(CO)ccc21 N1(C(C=CC=CCC)=O)CCC(C)(C)C(CNC(C2(NC(C)=O)CCC2)=O)C1 c1(C(=O)NC2CCN(C(C(C)(C)OC)=O)CC2C)c[nH]c2cnccc12 c1(C(N)=O)c(N2CCOCC(CNC(=O)Cc3ccco3)C2)ncnc1Cl c1(C(N)=O)cc(NC(=O)C(O)CC(F)(F)F)ccc1[N+](=O)[O-].C12CCN(C1)C2=O N1(C(C(C)N2CCC2)=O)CC2CC(C1)N(C(C13CCCC1C3(F)F)=O)C2 N1(C(c2c(CNC(C3NC(=O)CC(=O)C3)=O)occ2)=O)CCC2(CC1)CC2CO Cc1cc(C(F)(F)F)nc(N2CC(N(C)C(c3cccc(O)c3C)=O)C2)n1 c1(CC)ccc(C(=O)NCC2(F)CCN(C(=O)CCCN3CCCC3)C2)cc1Cl Cc1ccncc1CNC1CCC(C(=O)Nc2cccc(CO)n2)C1 C1(CNC(c2c(CNC(CCC3(C)N=N3)=O)ocn2)=O)COC(C)(C)CO1 N1(C(CCC2(C)CN(C(C3(COCC)CC(=C)C3)=O)C2)=O)CCC(O)C(F)(F)C1 CC1(C)C=C(C(=O)NC(CNC(c2ccn(C3CCCC3)n2)=O)CO)C1 C(=O)(C(=O)CC(C)C)N1C(CC)C(NC(=O)Cn2ccnc2C(C)C)CC1 C1(C(N2CC(C(C)C)C(C(=O)NCC(Cl)Cl)C2)=O)CN(C)CC(C)O1 N(C(=NCCc1cccs1)N1CCC(Oc2ccc(N)cc2)C1)C(C)CN(C)C CCCCC(C(=O)N1CCCN(C(c2cc3n(n2)CCOC3)=O)CC1C)C(C)C c1(OCC(N2CC(N(C(C(CC=CC)CC)=O)C)C2)=O)c(F)c(F)cc(F)c1F C=CCCCC(=O)NN1CCC(N(C)C(C2(Cc3ccc(O)cc3)CC2)=O)CC1 c1(C(=O)NC2(CNC(C3(O)CCSC3)=O)CC2)ccccc1SC(F)(F)F C1(NC(c2cc(C)n(C(F)F)n2)=O)CN(C(=O)C2=NOCC2)CC1N=[N+]=[N-] C1(C(N(C(C)C)CC)=O)CCCCN(C(=O)C=C(C2CC2)C2CC2)C1 O=C1CSc2ncnc(NC3CC(c4ccc(Cl)s4)C3)c2N1 O=C(N=c1cc(Cl)nc(Cl)[nH]1)C1CC(O)CN1Cc1ccncc1Br C(CC(F)F)(C(=O)N1CCOC(C2CC2)C1)N(C(=O)CC1OCCO1)C C(=O)(CC(F)(F)C(F)F)NCC1CCCN(C(c2c(C)n(C)cn2)=O)C1 CCC(C)C(C(=O)N1CC(C)C(C)(CNC(c2n[nH]cc2C)=O)C1)N(C)C C=CCCCCC(C(=O)NC1(C)CC1)N(CCCC(=O)NC)C CCCCCC(=O)NC1CC(F)(CNC(=O)CNC(=O)COc2ccccc2)C1 c1(CC)ncnc(NC2CC(NC(=O)Cc3cc(OC)no3)C2(C)C)c1F C=C1CCN(C(=O)CCC=CC(C)C)C(C(=O)NCC2CCNC(=O)C2)C1 C(CC(CC)C(=O)NC1CCC1C(F)F)=CC.c12ccc(cc1)OS(=O)(=O)N2 N1(C(CN2CCN(C(c3c(=O)ccn(C)c3)=O)CC2)=O)CC2(CCNC2=O)C1 C1(NC(CC(CC)OC)=O)C2CC3CN(C(C4C5CCC(F)(F)C45)=O)C1C3C2 Cc1cccc(-c2ccccc2CNc2cc(C(=O)Nc3ccno3)n(C)c2)c1 c1(OC)cc(CN2CCCC(C(=O)NC3(C)CCCCC3)C2)cc2c1OCO2 c1(OC)ccc(CC(=O)NCC(O)CN(C)C(C2CC2NC)=O)cc1F c1(OC)cccc(C(=O)NC(CNC(c2coc(O)n2)=O)C(C)(C)C)c1C C1(CNC(CC2C(C)C2)=O)COCCN1C(c1sc(=N)[nH]c1-c1ccccc1)=O C(=O)(CCCCCC#N)N(CC(C)O)CCNC(=O)CC1CCC(C)(C)CO1 c1(C(=O)NCC(CNC(C(C(C(C)C)O)C)=O)(C)C)cc(O)nc2c1CCCC2 N1(C(C(=O)NCCOCCOC)=O)CCCC(CCCC(=O)NC(C)(C)C)C1 C(=O)(C1=CCCO1)NCCC(CNC(C1CCCCN1C(C)C)=O)OC CC1(C)CC(C(=O)N2CCN(C(=O)CCCF)CC2C2CC2)c2ccccc2O1 N1(C(C(C(C)(C)C)SC)=O)CC2CCC1C(NC(c1csc(C(N)=O)n1)=O)C2 c1(C(=O)NC(CNC(COCC#C)=O)CO)cc2cc(Br)cnc2s1 C12(CNC(c3n(CC)cnn3)=O)CC1CN(C(=O)C(C)NC(=O)COC)C2 c1(C(N2C(C(C)NC(C3CCCC34CCC4)=O)CCC2)=O)ccc2c(c1)OCO2 c1(CNC(CNC(C)=O)=O)cccc(CN(C)C(c2cc(C)c(C)[nH]2)=O)c1 c1(OC)ccc2c(C(N3CC(C)(NC(c4cc(C)cnc4C)=O)C3)=O)csc2c1 CCCCC(O)Cc1nc(C(C)C)nn1-c1ccccc1OC c1(C(=O)NC2C3CC2N(C(=O)C=Cc2cccnc2)C3)ccnc2ncccc12 c1(C(N2CC(CC)(NC(=O)CO)C2)=O)cccc(CO)c1 C1(C)(CC)CC(C(N2CCOCC(CNC(c3cn(C)cn3)=O)C2)=O)CCO1 CN1CCN(C(C2C(NC(C3OC4CCC3C4)=O)C2(C)C)=O)CC12CCC2 C1(NC(C2(CC#C)CCOC2)=O)CN(C(=O)CCn2ccnn2)CC(F)(F)C1 N1(C(C(CC)SC)=O)CCCCCC1c1nc(-c2ccccc2)no1 C(=O)(CC(C)O)NCC(CC)N(C)C(c1nn[nH]n1)=O CC(C(=O)N1CC(O)CC1CC(=O)Nc1cnc(F)nc1)C(F)F CCC(F)(F)CC(=O)N1CC(CNC(=O)CCc2nc(C)no2)C(F)(CO)C1 Cc1ccc(CC(=O)NC2(CN(C(=O)CC3CCCCC3O)C)CC2)c(F)c1 C(=O)(C(CNC(=O)Cc1cc(C)cs1)C(C)(C)C)NCC(C)(CO)OC C(=O)(C(O)CC(N)=O)NC1CCC(NC(Cc2c(Br)cn(CC)n2)=O)C1 C(CC(O)CCO)NC(C1(CNC(Cn2ncc(C)c2)=O)CCCO1)=O N1(C(c2occ(C)c2)=O)CC(C)CCC1CNC(c1cc(C)cnc1N)=O C1(CC(=O)OC)CCC(C)N(N2CCCC(N3CCN(C(C)C)CC3)C2)C1 n1(CCC)ccc2cc(NC(C3CC(OC)CCO3)=O)ccc12 c1(NC(C2CCCN2C(C2CC(F)C2)=O)=O)ccc(Cn2ccnc2)cc1 Cc1ccc(-c2nc(C(=O)N(CC(C)(C)NC(C3C=CCCC3)=O)C)cs2)cn1 C1(NC(C2(CC=C)CCCCC2)=O)CCN(C(=O)CC(C)(C)C#N)CC1F N#CC1CN(Cc2ccc(O)c(Br)c2)CC1NC(c1csc(Cl)n1)=O CCCCC(C)CCC(=O)N1CCCC1C=CC(N1CCC1COC)=O N1(C(C(CC)C)=O)CC2(COC(CNC(=O)C=Cc3ccncc3C)C2)C1 CC1CCCc2c(C(N3CCCN(C(C4CC(F)C4)=O)CC3)=O)cnn21 C1(C(C)C)CN(C(=O)CC2CCC2)CCC1NC(c1ccn(C2CCC2)n1)=O C#Cc1ccccc1CC(=O)NC1(COC)CN(C(c2cccc(C#N)c2)=O)C1 N1(C(C2N(C(C(CC)(CC)CO)=O)C(C)C2)=O)CCOC2(CCCC2)C1 C1(C(NOCCOCC)=O)C2CC2CN1C(=O)C(C)n1ccnn1 C12(NC(=O)Cc3csc(Cl)c3)CCCN(C(=O)CCc3cscn3)CC1C2 CCCCC(COC)NC(=O)NC(c1cccc(F)c1)C1CCC1 C1(N(C(C(OC)OC)=O)CCO)CCCN(C(=O)CCc2ccc(O)nn2)C1 CC1CCCC(C)N1C(c1cncc(-c2ccc(O)cc2N(C)C)n1)=O CCCC(C(=O)N1CCC(N(c2ccc(Cl)cc2)CC2CC2)CC1)NC(N)=O c1(OC)cc(OC)nc(CN(c2nc(-c3ccccc3OC)cs2)C)n1 C1(C)(C(N(CCCNC(C=Cc2ccc(C)o2)=O)C)=O)CCC12CCC2 C(=O)(C(C)C(F)(F)F)NCC1CC(COC)CN1C(c1cscc1C)=O N1(C(CSCC(C)C)=O)CCOCC(C)(CNC(=O)C#CC2CC2)C1 c1(C(=O)OCC(=O)NC(C(CC)C)C)cccc(N2CCC(NC)C2)c1 CC(CC(=O)N1CC2CC1(C(=O)NC1C3CCC(F)(F)C13)C2)CC(C)(C)C c1(C(=O)NCC(CNC(c2cc(C)nc(O)c2)=O)(C)O)cc(F)cc(C)c1N N1(C(c2nc(N(C)C)oc2)=O)CCCCCC1C(N)=O Cc1cc(Cl)cc2[nH]c(C(=O)NCC3CCCN(C(=O)C(C)(Cl)Cl)C3)cc12 C1(C(N2CC=CC(NC(=O)CC3CC=CC3)C2)=O)CC2(C1)CS(=O)(=O)C2 CC1c2ccccc2OC1CNC(c1cc2c(Cl)cncc2s1)=O N#Cc1ccncc1C(=O)NC(c1ccc(Cl)cc1)C1(O)CCCC1 CC1CCN(C(=O)CCC2CCOCC2)CC1NC(C1(C)CCNC(=O)C1)=O N1(C(CC(C(C)C)O)=O)CC2C3CCC(C2C1)N(C(=O)CCc1ccc(Cl)s1)C3 C(C(C)CC(F)(F)F)NC(C1C(CC)CN(C(c2ccncc2O)=O)C1)=O CCC(C)CC(=O)NCCC1CCN(C(=O)CCOCC(F)F)CC1 C#Cc1ccc(C(N2CCCC2CC(N2CC3CC2CN3C)=O)=O)nc1 c1(CC)cc(C(=O)NCC(C)(O)CNC(C2CCC2C(=O)OC)=O)sc1C c1(CC(N2CC(CCCCNC(CCNC(COC)=O)=O)C2)=O)csc(C)n1 N#Cc1cccc(N(CCO)C(c2ccc(C3(F)CC3(F)F)cc2)=O)c1 C1(C(=O)NC(c2cnccn2)C)CN(C(c2cc(O)n(C)n2)=O)CC12CC2 c1(OC)ccc(CNC(c2c(CNC(=O)C(O)CSC)cnn2C)=O)nc1 C1(OC)CCN(C(=O)NCC2CC(F)(F)C2(C)C)C(C)(C)C1 c1(C(=O)NC(C(C)NC(c2cnc(C)[nH]2)=O)CO)ccc(F)c(C)c1C#N c1(C(N(C2CCN(C(c3cc(Cl)no3)=O)C2)CC)=O)csc(F)c1 C(=O)(CCCCCNC(C1(C)CCCN1C)=O)NCC(CC(=O)OC)O CCC(O)CC(=O)NCCc1ocnc1CNC(=O)CC(c1c(C)noc1C)C CCC(O)C(C)C(=O)NCC(C)(C)CC1CN(C(c2cc(Cl)n(C)n2)=O)C1 Cc1csc(S(=O)(=O)NC(C2CCN(C(c3ccncc3)=O)CC2)=O)c1 c1(C(=O)OC)cc(Br)c(C(=O)OCC2(C(F)(F)F)CC(O)C2)c(I)c1 c1(C(N2C(C)CC(NC(c3n(CC)ncc3)=O)C2)=O)cccc2c1CCC(=O)N2 N1(C(COC2CN(C(c3c(NC)cnnc3)=O)C2)=O)CCC2CCCC2CC1 c1(CC(=O)NC2CC(CNC(C3(C4CC4)CCCO3)=O)C2)nc(C(F)(F)F)cs1 N1(C(c2c(F)ncc(OC)c2)=O)CCCCCC(Nc2nc(C)nc(=N)[nH]2)C1 c1(N(C(C)(C)C)CCC#N)[nH]c(=NC2CCCC2C#N)ccc1[N+](=O)[O-] N1(C(C(C)(C2CCC2)NC(=O)C=CC2CCC2)=O)CC(CO)C2(CC2)C1 N1(C(CCSCCC)=O)CCC2CN(C(=O)C(CO)OC)CCC2C1 C#Cc1cccc(CNC(C2CC(C)N(CC)C2)=O)c1 Cc1nc2cncc(NC(C3CC3c3cc4ccccc4o3)=O)c2nc1C Cn1nnc2c1CCC(C(N1CCCC3(C1)CN(C(c1cc(F)cs1)=O)C3)=O)C2 C(CCCC(=O)N1CCC(C(C)CNC(c2oncc2C)=O)CC1)OCC c1(CCC(=O)NCCN(C)C(c2ccc(CSc3nc[nH]n3)o2)=O)c[nH]c(=N)[nH]1 C1(C(=O)NCCCCC=C)CCN(C(=O)C(=O)N(C)C)CCO1 c1(CC)cc(C(=O)NC(c2cccc(-c3nn[nH]n3)c2)C(F)(F)F)ccc1F N1(C(c2ccc(C)s2)=O)CCCC1C1CCCN1C(=O)COCCOCCO N1(C(C(CC)N2CCCC2=O)=O)CCCC(CN(C(=O)C(C(C)C)N(C)C)C)C1 CC(C(F)(F)C(F)(F)F)=CC(N1CC(C)CCC1CNC(c1csnc1C)=O)=O C(=O)(CC1=CCCC1)N1CC(CNC(CC(CC)C)=O)C1 C1(C(N(C)CCNC(=O)CS(=O)(=O)C2CC2)=O)CCC2(CC1)NC(=O)NC2=O c1(C(N2CC(O)(C(C)NC(C3CC(C(F)(F)F)CO3)=O)C2)=O)cccc(F)c1 C1(CNC(CCOCC#C)=O)CN(C(c2cc[nH]c2C)=O)CCC12CCOCC2 N1(C(c2c(C)cccc2)=O)CC2(C1)CN(C(C1CCCC(C(F)(F)F)C1)=O)C2 N1(C(C(CC)(C)C)=O)CCN(C)C(CNC(=O)C(c2ncccc2C)(F)F)C1 C1(CNC(N2CC(SC)CC2(C)C)=O)CC2(CCNCC2)CO1 C12(NC(c3ccc(CC)[nH]3)=O)CC(C)(C1)OC21CN(C(=O)C(C)(C)CC#N)C1 C(=O)(C(C)(O)C(C)C)NCC1(O)CN(C(c2ccc(SCC)nc2)=O)C1 Cc1nc2n(c1C(=O)Nc1cccc(-n3cnnn3)c1)CC(C)CC2 c1(CC(=O)NCC=CCNC(c2csc(Br)c2)=O)ccc(F)c(Cl)c1 CC1CCCCC1C(N1CC(NC(C2(c3cccc(Cl)n3)CC2)=O)C1)=O Cc1nc(S)nc(C)c1CCC(=O)NC(C)(CNC(C1CCC(=O)O1)=O)C(C)C CC1CCN(C(=O)CC(C)(C)CN(C)C)CC1NC(=O)C(C)(C)CN(C)C c1(C(=O)NC2CCCN(C(c3ccc(C4CC4)s3)=O)CC2)cnc2ncccn12 C(=O)(CCC1=NNC(=O)CC1)NCC1(OC)CCN(C(=O)CS(N)(=O)=O)CC1 C1(C(=O)NCC2(C)CC2)C=CC(NC(=O)Cn2cncn2)C1 c1(OCC)ccc(CC(N2CCC(C)C2CNC(=O)COC2CCC2)=O)nc1 N1(C(c2c(C(C)C)scn2)=O)CC(N(C)C(C2CCCCCC2)=O)C(F)C1 Cc1cc(C(=O)NC2(CNC(=O)CC(C)c3cccnc3)CC2)cnn1 O=S(=O)(C1CCCCC1)N1CCC(CS(=O)(=O)F)CC1 c1(C(=O)NC2(COC)CCN(C(=O)C(C)=C3CCCC3)C2)csc(S(C)(=O)=O)c1 c1(C(N2CCC(C(C)(C)C)(CNC(C3CCC3)=O)C2)=O)cnn2ccccc12 C1(NC(Cn2c(CCC)ncc2)=O)CS(=O)(=O)CC1NC(=O)C1=C(Cl)CCC1 N1(Cc2nnc(C)o2)CCC(C)C(NC(c2ccnc(C3CC3)c2)=O)C1 C(=O)(CS(=O)(=O)C1CC1)N1CC2CC(NC(c3nncc(C)c3)=O)C2C1 c1(OC)cc(C(N2CCC(C)(C(=O)N(C3CCN(C4CC4)C3)C)C2)=O)ccn1 CC1=C(C(=O)NCC2(O)CCN(C(=O)CN3CC4CC4C3)C2)C(C)(C)CCC1 c1(C(C)C(=O)NC2CCC2NC(=O)C(=Cc2c[nH]cn2)F)ccc(C2CC2)cc1 c1(CC)c(C(=O)N(C)CC2CC(F)CN2C(=O)C(O)C2CC2)cccc1F CC12CCCC(C(N3CC(C)N(C(=O)C(=O)N(C)C)CC3)=O)(CO1)C2.C1(N)CC1 C1(C(=O)NC(C)CCCNC(C2CCC2(F)F)=O)(OC)CCC(F)(F)CC1 C(c1csc(Br)c1)=CC(N1CC(N(C(C2C(OCC)C2)=O)C)C1)=O c1(CC)ccc(CC(=O)N(CCCNC(C2(C)CCCOC2)=O)C2CC2)cc1 N1(C(C(C)CF)=O)C(CNC(c2ccc(F)cc2F)=O)CC2COCC12 Cc1nccnc1C(=O)NC1CC2C(NC(C3(CCN=[N+]=[N-])CC3)=O)C2C1 c1(OC)cccc(C(=O)N(C2CN(C(c3cccc(N)c3)=O)CC2O)C)c1C N1(C(C2CN(C(C(CC#C)O)=O)CC2CC)=O)CCN(C)C(=O)C1CC c1(OCCCNc2nc(C)c(F)s2)ccc(F)c(Cl)c1 c1(OC)cc(C(=O)Nc2ccnc(O)c2)c(NC(c2ccc(C)cc2Br)=O)cn1 N1(C(CCCCCSC)=O)CCN(C(=O)C2=CC(C)(C)C2)CC(C)C1 Cc1ccc(C(C)NC(C2C3CC2N(C(c2cnc(C)c(C)c2)=O)C3)=O)cc1Cl n1(CC)nc(C)c(CC(=O)NCC2CCC(C)N(C(=O)CNS(N)(=O)=O)C2)c1C N1(C(C2(C#N)CCCO2)=O)CC2CCCN(C(c3csc4cncn34)=O)C2C1 c1(C(N2C(C(=O)NCCOCCOC)CCCC2)=O)ccc2[nH]nc(I)c2c1 C=CCCCC(=O)NC1CC1NC(=O)NCc1ccnc(Sc2ccccc2)c1 c1(NC(C)=O)cc(-c2cncnc2C(N2CCOCC2C(C)C)=O)cc(F)c1 n1(CC(=O)NCC2OCC(CNC(C)=O)C2)nc(C)n(C)c1=O C1(NC(C2CSCCS2)=O)CN(C(=O)CC2CCCC2(F)F)CC2(CCC2)C1 N1(C(c2n(C=C)ncc2)=O)CC2CCN(C(=O)CCc3scnc3C)CCC2C1 N1(C(CCC=CC)=O)CCN(C(=O)Cc2ccc(O)c(C)c2)CC1C(C)C Cc1n[nH]c(C)c1SCC(=O)NCC(O)CCNC(C1CCC1C(C)(C)C)=O c1(C(N(C2C3CN(C(=O)CCOCC4CC4)CC23)C)=O)sc2ccccc2c1Cl C1(C(N(C2CC2)CC)=O)CNCCN1Cc1cccc(-c2cccc(C)c2)c1 c1(C(N2CCC(CC(C)NC(C(C(C)O)C)=O)CC2)=O)ccc2ocnc2c1 c1(C(N(CCC(C)NC(C(C=C=C)C)=O)C)=O)cccc(N)c1NC c1(C(=O)NCCCCNC(c2ccc(C(C)=O)[nH]2)=O)ccc(OC(F)F)cn1 C1(CCC(=O)OC)CCCCN(C(=O)C(F)CC2CCOC2)C1.C12CCN1C2=O c1(CC(=O)NC2C3CCN(C(c4n(C=C)ncc4)=O)CC32)c[nH]c2ccncc12 C1(CNC(c2c(C)oc(C)c2C)=O)CN(C(C2(C)CCOCC2)=O)CC(C)(C)C1 c1(C(N2CCC(C(C)NC(C(CC)OC3CCCC3)=O)C2)=O)cccc(F)n1 C1(CC)CCCCN1C(=O)CC1CCN(C(C2SCC=C2C)=O)C1 CC1CC(NC(c2cc(O)ncn2)=O)CN1C(=O)C=CC=C(Cl)Cl Cc1ncnc2c1CC(C(=O)NC(C1(O)CN(C(=O)C3=COCC3)C1)C)CC2 C(=O)(C(C)(C)C(C)(F)F)NC1(CNC(C2CCN(C(C)=O)CC2)=O)CC(OC)C1 C#Cc1cnc(C(=O)N(C2CN(C(c3cc(CCC)on3)=O)CC2O)C)c(C)c1 N1(C(c2cnc(C(C)O)s2)=O)CC(C)CN(C(c2cc(N)nc(Cl)c2)=O)CC1C N1(Cc2ccc(CC(C)C)cc2)CC(C(=O)Nc2cocn2)CC(F)C1 C=Cc1ccc(N)cc1.c1(S)cccc(C#N)c1.N12CCOC(C1)CC1(CC1)C2=O CN1CCC(=CC(=O)NCC23CC2CN(C(c2cncc(O)c2)=O)C3)CC1 c1(SCC(N2CC(=Cc3cccc(F)c3)C2)=O)ccc2c(c1)CCC2 c1(OC(CNC(C(C)OC2CCCC2)=O)(C)C)ccc(F)cc1Cl.C1(=O)CO1 C1(NC(C(C)=C2CCCC2)=O)CN(C(=O)COC(C)C)CC1OC1CCCOC1 C#CC1(C(=O)N(CC(O)CNC(c2c[nH]nc2F)=O)C)CCCC1 C12(CNC(c3cnc(CC)s3)=O)CCCC1N(C(c1cccn1C)=O)CCC2 N1(C(c2c(C)ncs2)=O)CC2(C1)OC1(CNC(=O)COCCF)CC2(C(N)=O)C1 C1(CC)CN(C(C2(CO)CC2)=O)CCN1C(c1cc(Br)ccc1F)=O N1(C(C(C(C)C)n2cnnc2)=O)CC2CC1CN2C(c1ccc(Br)o1)=O Cc1coc(C(=O)N(CCNC(C2(Cc3ccccc3)COC2)=O)C(C)C)c1C CN1CCCC(C)(C(N2CC(CNC(=O)CSCC(F)F)C2)=O)C1 C1(OCCCC)CC(F)(F)CN1C(=O)CC1CCOC1=O C=C(Br)CC(C)(C)C(=O)NC1CC1CNC(=O)COCC(c1ccccc1)C c1(C(=O)NCC2CCN(C(c3c[nH]nc3Br)=O)C2)cccn2ccnc12 c1(OCCCC)ccc(C=CC(=O)N(CCCCNC(=O)C(C)O)C)cc1 C1(C(=O)NCC=CCNC(=O)C(C2CCCCC2)F)CN2CCC1(C)CC2 C12(F)CCN(CC1)C2.CC1(C)C(NC(c2cnn(CCF)c2)=O)C1C(F)F c1(CCCC)ccc(C=CC(N2CCC(C(=O)OC(=O)OCC)C2)=O)o1 C1(NC(CCCCOCC)=O)CC(CNC(c2cccc(CF)c2)=O)C12CCC2 c1(C(=O)NCCCC(C)NC(=O)CC(C)c2cnn(C)c2)nnc(O)cc1O N1(C(C(C)(F)F)=O)CCC2CC2(NC(c2ccc3cnoc3c2)=O)CC1 N1(C(c2c(C)c[nH]c2)=O)CCC2(CC1)CC2NC(c1cc(Cl)cnc1C)=O c1(C(N2CC(NC(c3ccco3)=O)CC(C)C2)=O)cccc2c1OCCN2 C1(C(N2CCCC(NC(=O)Cc3ccn(C(F)F)n3)C2)=O)CC(C2CC2)=NO1 C(c1cc(Br)ccc1OC)=CC(N1CCC(NC(CCCOCC)=O)C1)=O c1(OC)ccc2[nH]nc(C(=O)NC(C3CCN(C(C4(F)CC4)=O)C3)C)c2c1 c1(OC)cncc(C(=O)N(CCC(C)NC(c2cc(Cl)ccc2Cl)=O)C)c1C C(=O)(CC(F)(F)C(C)C)NC1CN(C(CCc2cnc(C)s2)=O)C(C)CC1 C#Cc1cccc(OCC(N2CCC(F)(CNC(=O)Cc3nncs3)CC2)=O)c1 C1(C(N(CCC(C(C)C)NC(C2(C)CCCO2)=O)C)=O)CN2CC3CC2(CO1)C3 N1(C(C(C=C=C)C)=O)CCN(C(=O)CN2CCCCCC2)C2CCCC12 C1(C(=O)NCCOCCCN(C(C(CC)OC)=O)C)CCc2c(ncn2C)C1 N1(C(C(C)O)=O)Cc2nccn2CC(NC(C2(C(=O)NCCO)CCC2)=O)C1 C1(C(=O)NCC=CCC(=O)NCCC2(C)CC2)COCOC1 N1(C(CCC2CC(OC)C2)=O)CC(=O)NCC1C(N1CCC(C)(CO)C1)=O C12(CC)CN(C(=O)CCc3ccc(O)cc3)C(CNC(=O)CC3(C)CC3F)(C1)C2 CN=c1ccc(C(=O)NC2C3CCC2N(C(C2CC(=O)N(C(C)C)C2)=O)C3)c[nH]1 C1(N)(C(=O)Nc2cncc(C(=O)OC)c2)CC[Si](C)(C)C1 N1(C(C#C)=O)CCCC2C1CCN2Cc1cc(OC)cc(F)c1 CC(C)CC(=O)N(CC(O)CN(C(=O)CN(CC(C)(C)C)C)C)C c1(C(N2CC(C(C(=O)NC(C(=O)N(CC)CC)C)OC)C2)=O)cccnc1S S(=O)(=O)(c1cccc(C(=O)Nc2ccc(Br)cc2F)c1)N(C(C)(C)CO)C C1(CNC(CCCc2onc(C)n2)=O)CC(F)CN1C(=O)C(F)C(C)C N1(C(COC2(C)CCCC2)=O)CC(=O)NCC1C(=O)NCCC1CCC1 N1(C(CCCOC(C)=O)=O)CC2(CCCC2)C1C(=O)NC1CCOCC1C c1(CC(C)C)cc(C(=O)NCC2CN(C(=O)CCC(=O)OC(C)(C)C)C2)n(C)n1 CC(C)CC(CC(=O)NC1CC(NC(=O)Cc2cncnc2O)C1)CC(N)=O CCC(C)C(O)C(C)C(=O)NC1(COC)CCN(C(=O)CCC(=O)N(C)CC)C1 C(C(C)(C)C1=CCCC1)NC(CC(C1CC1)NC(c1c(C)cc(O)nc1)=O)=O c1(C(N(C2CCN(C(C3CCOC3)=O)C2)CCC)=O)ccc(C2CC2)cc1 C1(CC)CCC(C(=O)NCc2ccc(C(=O)NCCC3CCOCC3)s2)O1 N1(C(C2C(C)OCCO2)=O)CCC2CN(C(C3CCSCC3)=O)CC2CC1 C1(CC)CC(C(N2CCN(C(C3CC(C)(C)CN3C)=O)C(CO)C2)=O)CC(=O)N1 C1(C(=O)NC2CC(CCC(=O)NCC3(C)CCCO3)C2)CC2(CCC2O)C1 c1(C(=O)NC2C(C(N3CCC(CC#C)CC3)=O)CCC2)cccc(C#N)c1C CC(CCCN=c1nc(CO)cc[nH]1)NC(=O)COC1CCCCC1C C1(C(=O)NCCN(OC)C)CN(C(c2ccc(Cl)cn2)=O)CC1C1CC1 c1(CNC(C(CC)C)(C)c2nnnn2CC2CC2)cnn2c1CCC2 N1(C(C2(C=C)CCC2)=O)CCC2CN(C(C3CC3C3CCC3)=O)C2C1 C1(C)(C(N(CCC(=O)NC2CC2)C)=O)CC(O)CN1C(=O)C(N)=O c1(CCC)cccc(-c2ccc(C(C)NC(C3C4CCC(C4)C3C)=O)cc2)c1O Cc1cc(CC(=O)NCc2csc(C(=O)NC(c3ccccn3)CO)c2)n(C)n1 C(=O)(CC(C)(C)C(F)F)Nc1c(C)cc(NC(c2cnc(Cl)s2)=O)cc1 c1(C(N2CCC(N(C(C=CC)=O)C)C(C)C2)=O)ccc2c(n1)NCC2 N1(C(C(=O)NCCC(=O)NC(c2nc[nH]n2)CC)C)CCCCC1 C12(C(N3CC(CC=C)(NC(=O)CCc4cnc(C)o4)C3)=O)CCCC1(C(N)=O)C2 N1(C(C(F)=C(C)C)=O)CCN(CCNC(c2ccnc(C3CCCC3)n2)=O)CC1 Cc1cc(Br)cc(F)c1NC(N1CC2COCC2(CO)C1)=O C1(NC(C(C)(C2CCC2)NC(=O)Cn2cc(C(F)F)cn2)=O)CCCCC1O N1(C(N2CCC(C)(C(=O)OC(C)(C)C)CC2)=O)CCC2(CC1)CC(O)CCO2 C1(SCC)N(C(=O)CSSC)CCC1(C)C.c12cccc(c1)NC(=O)C(CC)O2 N1(C(C(CCC)NC(=O)C(CCSC)NC(C)=O)=O)CCN(C)CC1CO C12(CC(=O)NC3C(NC(C(=O)NC(C)C)=O)CC3)CCC(CC1)C2 C1(CC(=O)NCC(C)CNC(c2cc(-c3ccco3)cs2)=O)OCCC1(C)C C(=O)(C1CCCn2cnnc21)NC1CCN(C(c2c(OC)scc2)=O)C12CC2 N1(C(C2(CC(C)C)CCC2)=O)CC2(C(=O)N(C)CC3CCCS3)CC1CO2 N1(C(CCC(CC)C)=O)CC(NC(C2CCN(C3CC3)CC2)=O)CC(F)(F)C1 Cc1cc(C(=O)NCCCOCCC(=O)NC2CCOC2(C)C)nnc1O c1(C(N2CC3C(NC(=O)C4=CCSC4)(C3)C2)=O)ccc2c(n1)CCC2=O CC(C)CCCC(=O)NCCC(C)N(C)C(c1ccc(-c2nccs2)cc1)=O O=C(C1=C(Cl)CCC1)NCC1(CO)CCN(C(C2CCC3(CCC3)C2)=O)CC1 C12(NC(c3cccc4[nH]ncc34)=O)CCCN(C(=O)C(O)C3CCC3)CC1C2 C1(C)(CC)CC(NC(c2occc2C2CC2)=O)CN1C(=O)Cn1cccnc1=O C(C)(C)(C(=O)NCCCN(C(=O)CCCn1cccc1)C(C)C)OCC C(CC1CCC1)(C(=O)N1CCCO1)NC(=O)CC1CCC=CCC1 N1(C(c2c(C)nc(N(C)C)s2)=O)CCN(C)CC1CNC(=O)C(C)c1cc[nH]n1 c1(C(N2C(CNC(C34CC(COC)(OC3)C4)=O)CC2)=O)cncc2ncn(C)c12 C(=O)(C1=CC=CN2CCS(=O)(=O)N=C12)NC(C)CNC(C1CCCC12CC2)=O c1(CC(=O)N(CCC)CCNC(=O)CC2C=NN(C)C2=O)cccc2ccoc12 c1(C(N2CCC(N(C(COC(CC)(C)C)=O)C)C2)=O)c(Cl)ccc(C)c1O N1(C(C(C)c2cccs2)=O)CCCC(CCNC(=O)CSc2ccncc2)C1 C(CC(C)(C)C(=O)NCC1(F)CCC(NC(C2CCC(=O)NC2)=O)C1)OC c1cc2c(NCCNC3CCOCC3)[nH]c(=NC3CC4(CC(C)C4)C3)nc2s1 c1(C(=O)NC2C(CNC(c3ccc(C4CC4)s3)=O)C2)cc2c([nH]1)CCCC2=O CS(=O)(=O)c1cncc(-c2cncnc2C(N2CC3CC3C2)=O)c1 C1(CNC(CC(c2cccc(C(F)(F)F)c2)C)=O)CCCC(CN=[N+]=[N-])C1 c1(C(N2C(C)CC(NC(=O)C(C3CCCCC3)O)C2)=O)cnc2c(c1)CCC2 CC(=NOCC#N)C(=O)NC1CC(CCC(=O)Nc2cnn(CC(C)C)c2)C1 n1(CC)nnc(C(=O)NCC(C)=CC(=O)NC(c2cnn(C)c2)CO)c1C C(C(O)C(F)F)NC(CCOCCN(C)C(c1cc(CCO)on1)=O)=O n1(CC(=O)NCC(CN(C(c2cn(CC)nn2)=O)C)O)ccc2cc(F)ccc12 C1(NC(c2n(CC)ncn2)=O)CN(C(c2cc(C)n(CC)n2)=O)CCC1C c1(C(=O)NC(C)CNC(=O)CSc2cn[nH]c2)csc(C(F)(F)F)n1 N1(C(Cc2cc(C)on2)=O)C2COCC1CC(NC(c1ncccc1C)=O)C2 C1(NCCC(CC)C)CCOC(c2ccc(F)cc2)C1 C(=O)(C(C)(O)CC(F)F)NC1CCC(NC(C=Cc2cncc(C)c2)=O)CC1 C(=O)(CCN=c1[nH]c(=NCc2ccc(Br)cc2Cl)[nH]c2c1SCC2)NC CCC(C(=O)NCC(c1ccccc1CO)NC(c1c(C)cnn1C)=O)C(C)O C1(N(C)C(=O)NC(C)(C)C)CN(C(=O)OC(C)(C)C)CCC12CCOCC2 c1(CNC(C(=O)NCCN2CCOCC2)CC2CCC2)ncc2ccccc2n1 C12(CNC(=O)COCC(F)(F)F)CCCCC1CN(C(c1csnn1)=O)C2 C1(C2C(c3c(C)cco3)C2)CCC2(CC1)CNC2.c1(C)cnc(C2CC2)o1 N1(C(C2(CC)CN(C(=O)CC3(C#N)CC3)C2)=O)CCC(C)(C)C1C c1(C(=O)OC)ccc(O)nc1NCC1C2CN(C(c3cc(=O)cc(Cl)[nH]3)=O)CC12 N1(C(C(=O)NCCCCCC)C2CC2(C)Br)CCC(O)(CCC)CC1 N1(C(CC(C)N(C)C)=O)CCC2(CCC2NC(c2cnc3ccnn3c2)=O)CC1 c1(C(=O)NC2CC(C(=O)Nc3cnc(C(=O)OCC)s3)C2)c(I)ccnc1F C(=O)(C#CC(C)(C)O)NCc1cc(C(=O)NCC(CC(C)C)N(C)C)n[nH]1 C(=O)(CCCCC(=O)N1CCCC1CCNC(=O)Cc1conc1C)OC Cc1cc(C)c(C(N2CCN(C(c3cc(Cl)c[nH]3)=O)C(C(C)(C)C)C2)=O)cc1C CC1(C(N2CC(NC(=O)CSc3cn[nH]c3)C(C(F)F)C2)=O)CC=CCC1 c1(C(N(C)CC2(NC(=O)CCCN3CCOC3=O)CC2)=O)cnc(C2CC2)s1 S(=O)(=O)(c1ccc2cc(Cl)sc2c1)N1CCN(c2cc(C)nc(C)n2)CC1 Cc1cc(NC(=O)NC(C)CN(CCC(F)(F)F)C)cc([N+](=O)[O-])c1 CN1N=C(CC(=O)N2CCC2CC(N2CC(CO)CC2(C)C)=O)CC1=O C1(CSC)NC(=O)N(CC(C)(C)CN2CCOCC2)C1=O CC1COCC(CNCCn2cc(CNC(=O)CNc3ccccc3Cl)nn2)O1 CCCS(=O)(=O)C(C)C(=O)NC1(C2CCN(C(C3(CO)CC3)=O)CC2)CC1 N1(C(C(C)OCCCCCC)=O)Cc2[nH]nc(C(=O)NC(C)CO)c2C1 N1(C(CN(C(C)C)C)=O)CCC(CC(N)=O)(NC(C2CCC(F)CC2)=O)CC1 C(CC(=O)N1CC(CCNC(c2cn[nH]c2)=O)C(C)C1)(C(N)=O)NC(C)=O c1(C(N(C2CN(C(C(CC)(C)C)=O)CC23CC3)C)=O)ccc2[nH]c(C)c(C)c2c1 CC(C)C(CC(=O)NCC(C)CO)NC(=O)CCCn1cccn1 n1(CC(N2CCC(NC(C)C)CC2)=O)cnc2c1CCCC2 C1(Oc2ccc(-c3nncc(C)c3C)cc2)CC(C2CCCC2)C1 N1(C(=O)CCc2nccs2)CC2CN(C(C3CC3Br)=O)CC2C1 N(C(=NCc1ccn(C)n1)NC1CCOCC1)C(C)C1CC1 c1(C(N(C(C)CNC(c2nccc(C(F)(F)F)n2)=O)CC)=O)cn(C)[nH]c1=N C1(C(=O)NCC(C)NC(C(C2CCOCC2)OCC)=O)CC(=O)NC(=O)N1 c1(CC(N2CCN(Cc3nc(C)on3)CC2)=O)cn2cc(C(F)(F)F)ccc2n1 c1(OCC=C)ccccc1C(=O)NC(CNC(C1CCCC1CC)=O)C(C)(C)C C1(CNC(C(c2ccc(OC)cc2)C)=O)C(C2CC2)CCN1c1ncncc1Cl C12(CCNC(c3nnc(C)s3)=O)CCC1CN(C(c1cc(Cl)ccc1O)=O)C2 Cc1cccc(F)c1C(=O)NC1CCN(C(=O)CC2(N(C)C)CCCC2)C1C CC1C=C(C(=O)NCc2ccc(CN(C)C(C34CCC(C3)C4)=O)cc2)C1 C1(n2c(-c3nc(Cl)oc3C)nc(CCOC)n2)CCCCC1(C)C c1(CCC(N2C(CNC(=O)CCc3ncc[nH]3)CC2)=O)cccnc1Br c1(C(N(C2CCCN(C(=O)C=Cc3scnc3C)C2)CC)=O)ccnc(NC)c1 C12(CC(=O)NCC3CCCN3C(=O)C(C3CCCCC3)O)CCC(CC1)OC2 N1(C(c2c(CC)nn[nH]2)=O)CC(CNC(=O)C(C)N2CCC2)CC(C)(C)C1 C1(NC(c2cc(C)sn2)=O)CC2CCC1C(NC(=O)CC1CCCC3(CC3)C1)C2 C12(NC(C(C(C)O)C)=O)CC(CNC(c3cc(Cl)cc(Cl)c3)=O)(C1)OC2C Cc1cccc(CC2CCN(C(=O)NCCC34CC(CO3)C4)C2)c1F C1(CC(=O)NCC2(O)CN(C)C2)(OC)CN(C(=O)C(c2ccccc2)O)C1 c1(C(C)Cn2cc(CN3CCC(CN4CCCC4)C3)nn2)ccc(C#N)cc1 C#Cc1cnn(CC(N2CCC2(C)CC(=O)NCC(O)CCOC)=O)c1 c1(CC)cc(C(=O)NCC(CO)NC(=O)CCc2cnc[nH]2)ccc1C c1(C(=O)NC2C(CC)CN(C(=O)CCCC(C)C)CC2)cn2ncnc2nc1C N1(C(C(C)n2ccnc2)=O)CCC(C(=O)N2CCC(C)(F)CC2)=C(F)C1 C1(C(=O)NC2(C)CSC2)CN(C(c2ccc(F)cc2F)=O)CC12CC2 Cc1cc(Br)c(CC(=O)NC2CCC(CNC(c3sccc3F)=O)C2)s1 C1(C(=O)NC(CC)C2CC2)CC(C)CCN1C(=O)C(O)CSC c1(OC)ccc2[nH]nc(C(=O)NC3CC(C)N(C(=O)CC(C)(C)F)C3)c2c1 C(=O)(CC1=CCOCC1)N(C(C)(C)CC(N1CCCC(C(F)F)C1)=O)C c1(CC)cc(C(=O)NC2(C)CC(NC(=O)CC3CCOCC3OC)C2)nn1C CC1(CNC(C2CC2Br)=O)CCCN1C(c1ccc(-n2ccnc2)cc1)=O N1(C(CC2(C)CCOCC2)=O)CC2CC(C(N3CCCC(F)(CO)C3)=O)C(C2)C1 N1(C(CN(CC)CC)=O)Cc2ccccc2CC1CNC(c1cnc(C)[nH]1)=O C1(CN(C(=O)C(C)(C)CF)C)CCCN(C(C2C(Cl)(Cl)C23CC3)=O)C1 c1(NC(C2(C)CC2)CO)cccc(Br)c1.C1CC(=O)OCC(=O)N1 c1(CSCC)ccc(C(=O)NCCN(C(=O)CCCc2cc(C)sc2C)C)cc1 c1(NCc2cn(CC(=O)NCCOCC(=C)C)nn2)ccc(F)cc1C C(CCCCC(=O)NCCCSC)N(C(c1c(CCC)n[nH]c1)=O)C c1(C(C(=O)N(C(CN(C(C=CC=CC)=O)C)C)C)OC(C)C)ccccc1 c1(C(C)(C)OC)nc(=NCCC2CCCCN2C(C2CC2(C)C(C)C)=O)s[nH]1 C1(O)(C(=O)NCCCOCCNC(CC(C(=C)C)O)=O)CCCC(C)(C)C1 c1(C(=O)NCCn2cc(C3(C(=O)OCC)CCC3)nn2)cc(C)cnc1F N1(C(CC(COC)(C)O)=O)CCC2(CC1)CC2NC(c1csc(C(N)=O)n1)=O c1(C(=O)NC2(CNC(CCCC(OC)OC)=O)CCC2)ncnc2sccc12 C1(CNC(C(C)N(C)C)=O)(CNC(c2ccns2)=O)CC(F)(F)C1 N1(C(c2cnc(C)s2)=O)CCCC(N(C(=O)C2=CCSC2)C)C1 Cc1ccc(C(=O)Nc2cccc(-c3nnnn3C)c2)c(Cl)c1 c1(OC)ccc(C)cc1NC(=O)CNC1CN(C(=O)Cn2cccc2)CC1(F)F N1(C2CC3CN(C(=O)Cc4cc(F)ccc4F)C2C3)CCOC2COCC2C1 N1(C(CCOCC)=O)CCC2C(CCCN2c2nc3ccccc3s2)C1 CC1(C)CCC(CNC(=O)C(c2ccco2)NC(=O)C(=O)N(C)C)O1 C1(NC(C(=C(C)C2CC2)F)=O)CCN(C(=O)Cc2c(Br)cnn2C)CC1 C1(C(N2C3C(CNC(=O)CN4CCCCCC4)C(C3)C2)=O)SC2C=CC1CC2 N1(C(c2cc(CC)on2)=O)CCC(NC(=O)C(c2c(C)n[nH]c2C)C)C(F)C1 CN=c1[nH]c(=NCC2CCCC23CC3)[nH]c(=NC(C)c2ccoc2)[nH]1 Cc1ccc(N(C)C(C2C3CN(C(c4ccns4)=O)CC23)=O)c(C)c1 N1(C(C(CCC)(C)C)=O)CCCC(C2CCN(C(C3(CO)CCCC3)=O)CC2)C1 c1(C(=O)NC(CC(C)NC(c2ccc(F)cc2)=O)C)ccc2nnn(C)c2c1 C#Cc1cc(C(=O)NC(C2CCCN2C(C2CCCN2C(C)=O)=O)C)ccc1Cl N(C1CCCn2nccc21)CCCCc1ccc(C(C)(C)C)cc1 C1(CCC)NCCN(C(=O)OC(C)(C)C)C1C(=O)OCc1nc(C(C)(C)O)n[nH]1 CON1CCC(CC(=O)NC2CC(CCNC(c3nc(C)no3)=O)C2)CC1 Cc1cc(CCC(=O)NC2CN(C(=O)COc3ccc(Cl)cc3)C2)nn1C c1(C(C)C)[nH]nc2cncc(C(=O)NC(C)CC(C)NC(=O)C(C)(O)C(C)C)c12 CCC(F)(F)CC(=O)NCc1occc1C(=O)N(C)Cc1cncnc1 c1(C(C)C)ccc(C(=O)NC(CNC(=O)CCOCC(F)(F)F)C(C)C)cc1Cl CCCCCC(=O)NCC1CC(F)(CNC(c2ccc(C(F)(F)CF)cc2)=O)C1 c1(C(=O)NCCCNC(C(COCC)C)=O)ccc(OC)c(C)c1OC CC(CS(C)=O)C(=O)NC1CC(NC(=O)CNC(=O)Nc2ccccc2)C1 N1(CCCc2ccccc2)CCN(N2CCN(Cc3ccc(Cl)cc3)CC2)CC1 C1(C(=O)NCc2ncc(OC)nc2)CC(=O)OC12CCCCC2 c1(NC2CC(NC(CCCNS(C)(=O)=O)=O)C2(C)C)ccc(C#N)cc1[N+](=O)[O-] N1(C(CC(C=C)CC)=O)CCCCC1C1CCCN1C(C1CCCCC1OC)=O C1(C(N2CC(CCNC(C=C(C)C)=O)OC(C)C2)=O)CC2C=CC1C21CC1 C1(CNC(COC(C)=O)=O)CC2CCC1N(C(c1cn(C(C)C)nc1C)=O)C2 CC1CCN(C(=O)C(C(C)(C)C)C2CCCCC2)CC1(F)F c1(C(=O)NCC2CC(NC(C3CCCC3n3cccc3)=O)C2)coc(C(F)F)c1 C1(CC=C(C)C)CCC(C(=O)N(CC(C)(C)C)CCCN(C)C)CC1.C1CO1 C1(C2CCN(C(c3ccn4nccc4c3)=O)C2)(NC(c2nncs2)=O)CC1 Cc1ccc(C)c(-c2nc(Cc3ccc(C)nc3)nn2C(c2cnn(C)c2)C)n1 N1(Cc2cn(CC3N(C(C)=O)CCC3)nn2)CCOC2(CCN(C)C2)C1 c1(-c2ccc(C)cc2)ccc(C(=O)O)cc1NCCN1CCCC1C N1(C(C)=O)CC(NC(=O)Nc2cnc(N3CCOCC3)nc2C)CC(O)C1 c1(OC)cc(CN2CCOCC2C(=O)Nc2ccccc2C(N)=O)cc(Cl)c1O C(CCC(C)C)(C(=O)NC(CCF)C(=O)OC)NC(c1c(CC)occ1)=O C=CCC(CC(C)C)C(=O)N1CCN(C(C2CC(OC)C2)=O)C(CO)C1 C1(COC)CN(C(c2ccc(C(F)F)o2)=O)CCN1C(=O)CN1CCCCC1 c1(NC)cnc(Cl)cc1C(N1CCCC1CCNC(=O)CC1CN(C)C1)=O CC(C)CC(C)C(=O)NCCCCCC1CCN(C(=O)C#CC(C)(C)C)CC1 Cc1cnc(C(=O)NCC(O)CCNC(=O)CNc2ccccn2)cc1C c1(CC(=O)NCCCCNC(C2(C(N)=O)CC2)=O)cccc2nonc12 Cc1cc(C(=O)NC2CCC(C)N(C(=O)COc3ccccc3)C2)cc(N)c1Cl c1(C(=O)NC2C(C)CN(C(c3c[nH]cc3Br)=O)C2)cc2ccc(F)cc2[nH]1 C=CC(CCC)CC(=O)NCC1CCCCN(C(=O)C=Cc2ccsc2)CC1 C=CC(C)(C)CC(=O)N1CCC1CC(N1CCOC(C(=O)OC)C1)=O C(N=c1[nH]c(=NCCN2CCC(C)CC2)[nH]c2c1CCC2)C1CCC(CC)O1 c1(C(=O)NCCC(CNC(c2c(C)ncn2C)=O)O)ccc2c(c1)NC(=O)CO2 C1(C)(C(N2C(C)(C(C)C)CC2)=O)CCN(C(=O)C=Cc2cnccn2)C1 c1(COC)cccc(C(N2CCC(NC(=O)C3CC3)C(C)C2)=O)c1C Cc1cnc(N(CC(=O)N)C)[nH]1.C1(N(C(C)(C)C)CC2CC2)CCN(C(N)=O)C1 CC1CN2CCN1C(C(=O)NC1CC1C1CCN(C(=O)Cc3ccsn3)CC1)C2 C1(C(=O)NC(CNC(C2(O)CCCC2)=O)CO)CSc2ccccc2O1 S(=O)(=O)(c1ccc(C#N)c(NCCC2COC(C)(C)O2)c1)NCC(COCC)C C1(NC(=O)C(O)Cn2cncn2)CC2CC(NC(C3C4CCCCC34)=O)C2C1 C1(CNC(CCc2cnc(C)o2)=O)CCN(C(c2c(C)nn(C)c2C)=O)CC1C C1(N(C(=O)C2=NOCC2)CC)CCCN(C(c2ccc(C(C)C)o2)=O)CC1 C(C(C)(CC(C)C)NC(=O)Cn1cnnn1)NC(c1cccc(SCCC)c1)=O N1(C(CC2C(C)C2)=O)CCN(CCN(C(=O)Cc2nc(C3CC3)nn2C)C)CC1 c1(CC(N2CC(CC(C)NC(C3C(C(=O)OC)C3)=O)C2)=O)cc(Cl)cs1 N1(C(C(C)Sc2ccc(N)cc2)=O)CCC(C)(C)C(NC(=O)CCC2(C)CC2)C1 n1(-c2cn(CC)nc2)nc(C2CCCCC2)nc1-n1ccc(C)n1 CC(C)(C)CC(F)C(=O)NCCCN(C1CCCC1)C(C1C(C(F)F)C1(C)C)=O N(C(=NCCSC)NCC(c1c(O)cccc1F)O)CC(c1scc(C)n1)C CC(C)C1=NOC(C(N2CCCCC2CC(=O)NCC2(N(C)C)CCC2)=O)C1 C1(NC(CSCC=C)=O)COC2CN(C(c3nc(Cl)ccc3N)=O)CC12 c1(C(=O)NCC(CN(C(C2(OC)CC2)=O)C)C)cnc2ccc(C)cn12 C(=O)(C(C(C)CC)NC(C1CC(C)(C)CO1)=O)NCCCC O=C(CCc1nncs1)NC1CC1NC(C1(C(N)=O)CC1)=O C1(CNC(C2(C(=O)Nc3cnc4snnc4c3)CC2)=O)COC2(CCNCC2)C1 c1(C(=O)NC2C(NC(C3(CCOC)CCC3)=O)CC2)cc2ccccc2c(O)n1 N1(C(C2(CC)CCC2)=O)CCC(O)(CNC(C2CCCN(CC(F)F)C2)=O)CC1 c1(CC)nnsc1CNC(=O)C(C)=CCNC(=O)C(CO)OC c1(C(=O)NCCCC2(NC(CCc3scc(C)n3)=O)CCC2)cccc(CF)c1 C#CC1(C(=O)NC(CC(=O)NCc2cc(C(C)C)no2)C(F)F)CCCCC1 N1(C(C(N2CCCC(C)C2)=O)=O)CCCN(C(=O)C(C)(C)c2cnco2)CC1 C(CC(C(C)(C)C)NC(C1COCCN1C1CCCC1)=O)N(C)C(c1cscn1)=O N1(C(CCNC(C)=O)=O)CCN(C(=O)CC2COCCO2)CC(C)C1 Nc1ccc(C(=O)NC2CCCCC2NC(C2CC3C(C2)C3(F)F)=O)nc1F c1(SC)cccnc1C(N1CCC(CO)(NC(C2CCC23CCC3)=O)C1)=O C(=O)(C(O)CC(N)=O)NC1C(C)N(C(=O)CN(c2ccccc2)C)CC1 N1(C(=O)CSCc2cccs2)CCC(c2cn(CCO)nn2)C1 C1(NC(c2cnn(-c3ccncc3)c2)=O)C=CCN(C(C2(O)CC2)=O)C1 N1(C(c2c(OC)ccnc2F)=O)CCCN(C(=O)C(O)C(F)(F)F)CCC1 C1(N(C(=O)CNc2ccccc2Cl)C)CCN(C(c2ccnnc2)=O)CC12CC2 C1(C(N2CCC(N(C34CC(C3)C(C)O4)C(C)=O)CC2)=O)CCC2CCC(=O)N12 C1(C(=O)NC2C=CCN(C(c3cnccn3)=O)C2)CC12CC(F)(F)C2 N#Cc1cc(NC(C2CN(C(c3cc(Cl)cnc3Br)=O)CCC2O)=O)cnc1Cl c1(C(=O)NC2(C3N(C(C(CC)COC)=O)CCC3)CC2)cc(O)nc(Cl)c1 C1(NC(COCCCC#C)=O)CCCCC1CNC(c1cc(COC)cs1)=O N1(C(c2n(C)ncc2C#N)=O)CC2(CCN(C(=O)C3=CCOCC3)C2)C1 C1(NC(c2cc(C(C)(F)F)n[nH]2)=O)CC1C1CCN(C(c2sccc2Cl)=O)CC1 c1(CN2CCC(C)(C(=O)N(CCCO)CCCO)C2)cc(Cl)nc(Cl)c1 c1(NC(CN2CC(Oc3c(C)occc3=O)C2)=O)cnn2ccc(O)nc12 C#Cc1ccc(CC(=O)NC(CNC(C2CC(C)(C)CCO2)=O)C2CC2)cc1 N1(C(C2(C)CC2(F)Cl)=O)CCC(F)(CNC(=O)Cn2ccc(C(F)(F)F)n2)CC1 Cc1sc(CC(F)(F)F)nc1C(=O)NCCCN(C(C1(O)CCOC1)=O)C1CC1 C=C(CNC(c1c[nH]nc1C)=O)CCNC(c1[nH]nnc1-c1ccnn1C)=O c1(C(=O)NCC2COCCN(C(C(F)OC)=O)C2)cc([N+](=O)[O-])cc(C)n1 N1(C(=O)OC(C)(C)C)CC2CC(C(=O)Cn3cc(-c4n[nH]cc4[N+](=O)[O-])nn3)C1C2 C1(NC(c2nc(CN(C(CCOC)=O)C)oc2)=O)CC=C(C(C)C)CC1 CC1CC(C(N2CCC(F)(C(N)=O)C2)=O)CCN1C(C1CN(C(N)=O)C1)=O S(=O)(=O)(c1ccc(F)cc1)N(CC(=O)N(C)CCN(C(=O)CC1CC(=O)C1)C)C C1(C(=O)NC(CCC)CCO)CC12CCN(Cc1ccc(N(C)C)c(Br)c1)C2 C(=O)(CCCC(C)O)NCCCOCC(C)(C)NC(c1nc(CC)sc1)=O c1(C(=O)NCCN(CC(C)O)C(=O)Cc2ccnn2C)ccccc1-n1cccc1 c1(C(=O)NC2C3CN(C(CCCSC)=O)CC2C3)cc2cc[nH]c(=O)c2s1 c1(N(C(C)CCNC(c2ccc3nonc3c2)=O)C)[nH]cnc2nc(Cl)cc1-2 C1(C(C)NC(C(C)=CC2CC2)=O)CN(C(=O)CC2(C)CC2)CCO1 C1(CN(C)Cc2ncccc2Cl)CN2CCCCC2CO1 C1(CC(=O)NCC(COC)(F)F)CC(NC(C2CC(=O)C2)=O)CCO1 c1(C(N(C)CCNC(C2(Oc3ccc(F)cc3)CC2)=O)=O)cc(F)ccc1Cl c1(CCCC(=O)NC(c2ccc(F)cc2)CO)cccc(Br)c1 C=CCC(CC(C)C)C(=O)NC1(C)CCC(NC(c2c[nH]nc2CCC)=O)CC1 C1(CC(=O)NCCC(C)N(C)C)C2CCCC2N1C(=O)CC(F)(F)F c1(OC)cccc(NC(c2c(OC)cccc2O)=O)c1Cl C1(C(C)C)CCC(C(=O)NCCOCCCNC(=O)CCN(C)C)C(=O)N1 CCC(C)C(=O)NCC(=O)N(C(CNC(=O)C(F)(F)C12CC(C1)C2)C(C)C)CC Cc1ccc(F)cc1CC(=O)NCCC1(O)CN(C(C2CCC(C)O2)=O)C1 c1(C(=O)OCC)ccccc1C(=O)NC(C1(CNC(=O)C(C)O)CC1)C C(CO)(CCCO)SC(C)C.C1CCC(=O)NC(C)C(=O)NC12CCC2 N1(C(c2c(C)nc(C)o2)=O)CCN(C(=O)Cc2ccoc2C)C(C(C)(C)C)C1 Cc1cnnc(O)c1C(=O)NCC1CCC1NC(=O)CC1COCC(C)(C)O1 c1(OCOC)ccc(CN2CCC(F)(C(N3CCC(C(=O)OC)C3)=O)C2)cc1 c1(C(=O)NC2C(NC(CCC(=O)NCCC)=O)C2)nnc2ccccc2c1O C1(NC(C2(NC(C3COCCO3)=O)CCCC2)=O)CCC2(CC2)C1 C1(C(C)C)(C(=O)NC2CC2NC(c2cn(C(F)F)cn2)=O)CNC(=O)C1 C(=O)(CC(O)C(C)C)N(CCOCCNC(C1CC=C(C)CC1)=O)C C1(CCNC(C2N(CC)CCOC2)=O)CC(F)(F)CN1C(=O)CN(S(C)(=O)=O)C CCC(CC)CCCC(=O)NC1CC(N(C)C(c2ccc3ccccc3c2)=O)C1 C(=O)(CCCC(F)F)N(C)CC1(O)CCN(C(c2c(CC(C)C)nc(C)s2)=O)C1 C=C(Cl)CCC(=O)N1CC(NC(=O)CCC(C)c2ccccc2)C(C)C1 C1(CNC(C(C)=C(C)C)=O)CN(C(C2(CO)CCCC2)=O)CC1(F)F CC1CC(N(C)C(=O)NCC2CCCC(=O)N2)CCO1 O=C1CC(C(=O)NCCc2nccc(O)n2)N(C(C2CCCC(=O)N2)=O)C1 C1(CC(N2C(CNC(CC3(CSC)CC3)=O)CC2)=O)COc2ccccc2O1 C1(NC(C(C)OCC)=O)CCN(CC(=O)Nc2ccc(F)cc2)CC1O C1(CC)CN(C(C2CCSCC2)=O)CCC1NC(c1ccc(CC(N)=O)cc1)=O c1(C(N2CCCC(c3ncn(C)n3)C2)=O)nc[nH]c1[N+](=O)[O-] C1(OC)CN(C(C2CCOCC2)=O)CC1NC(C1CC2(CC2)CO1)=O C1(OC)CN2C(=O)N(Cc3cc(C#N)ccc3Cl)C(=O)C2(C)C1 N(C(=NCC1CC1)NC1CCCN(c2ccccn2)C1)C(c1ccsc1Br)C N1(C(=O)OCC)CCC(NCCC(C)N(C)Cc2cn(CC(=O)N(C)C)nn2)C1 C12CC(C1)CCCNC2=O.C=CCCC1(CN)CC1.C(C)(=O)O Cc1cccc(C(=O)NCC2(CO)CCN(C(C3CCCS3)=O)C2)c1C C1(CCNC(C2C(COC)CC2)=O)CC(OC)CN1C(=O)CNC(=O)NC CN1C(=O)C(=O)N(CC(N2CC(CCNC(c3occc3C3CC3)=O)C2)=O)C1=O C(c1cc(C)cc(C)c1)=CC(=O)NCC1C2N(C(C(C(=C)Cl)(C)C)=O)C(CC2)C1 c1(CNC(CC2(NC)CC2)=O)cn(CC(N2CCCC2c2cccnc2)=O)nn1 C1(C(=O)NC(CC=C)CNC(c2c(Cl)cnn2C(C)C)=O)CCN(OC)CC1 C1(CC(=O)NCCC(Cn2cc(CCCOC)nn2)F)CCCC(C#N)C1 c1(C(=O)OC)cccc(C(C)=Cc2cccc(C(F)F)c2)c1 N1(C(C=CCC)=O)CC2CCN(C(C3(C)CC=CCC3)=O)CC2C1 c1(C(=O)NC2(C(F)(F)F)CCN(C(=O)CO)C2)cccc2c1OC(F)(F)O2 c1(CC)cc(C(N2CCCC(C)(CNC(C3CC(F)(CO)C3)=O)C2)=O)cc(Cl)n1 C1(NC(C(F)=CCC)=O)CCOC12CCN(C(=O)CC1CCCC(OC)C1)CC2 C1(C(N2C(C3(C(N4CC(C(N(C)C)=O)C4)=O)CC3)CCC2)=O)OCCCC1(C)C c1(CN2CC(C(=O)Nc3cncc(C)n3)OCC2)cn(C)c2ncccc12 CS(=O)CCC(=O)NCCCCCC(C)C.c1(C(=O)N)ccccc1CC(=O)O C(=O)(CC(C(F)F)C(C)(C)C)NCCCN(C(c1cc(C)c(C)o1)=O)C1CC1 N1(C(CCNS(CC)(=O)=O)=O)CCN(C(c2cc(F)cc(Cl)c2)=O)C2CC12 C1(NC(c2cc(C)on2)=O)CN(C(c2cccc(F)c2N)=O)C2CCCCC12 N1(C(C2N(C)CC(F)C2)=O)CCOCC(F)(CNC(=O)COC2CCCC2)C1 C1(CNC(COCC(C)C)=O)CCC(C)CN1C(c1ccc(C2(C)CC2)cc1)=O CC1(C)CN(C(=O)C(C2(C)CC2)NC(c2ccc(F)c(F)c2)=O)CCS1 N1(C(C(C)NC(C2CCC2)=O)=O)CCC2(CC(NC(C3(F)CCCCC3)=O)C2)C1 C1(C(=O)NCC(Cl)=CCl)(COC)C=CCN1C(=O)CCn1ccnc1 c1(C(=O)NC(CC)CNC(C2CCCN2C)=O)ccc(OCCF)cc1F CC1(F)CC2(CN(C(C3c4cn(nn4)C4N3CCC4)=O)C2)C1.C1COC1.NC=O N1(C(C=CCOC)=O)CCN(CC(=O)NCc2ncoc2C)CC1 c1(OCC)ccc(C(CO)NC(c2ccc(C)nn2)=O)cc1 C12(C(=O)NC3CC(C)(NC(c4c(C)ccc(C)c4)=O)C3)CCC(=O)N1CCS2 CC(CN1CCC(Cc2ccc(F)cc2)C1)CC(C)(C)C N1(C(CCC#C)=O)CC(C)OC2(CCN(C(=O)CCCC(=O)N(C)C)C2)C1 c1(C(=O)NC(CC#C)CC(=O)OC)c(C)sc2c(Br)cccc12 c1(C(=O)OC)ccc(NC(C2CCN(Cc3cncc(Cl)c3)CC2O)=O)cc1I N1(C(C(C)NC(C)=O)=O)CCC(C)(C)C1CC(=O)NCC1(O)CCCCC1 O=C(C1=COc2ccccc2O1)NC1C=CCN(C(C2C3CCC(F)(F)C23)=O)C1 C1(C(N(CCC(C(C)C)NC(C(CC#C)C)=O)C)=O)CCn2c(C)cnc2C1 c1(C(=O)NC2CC(CNC(C(c3ccc(C)cc3)C)=O)C2)cc2oc(C)cc2[nH]1 S(=O)(=O)(CCCN1CCCC1=O)NC(c1cc(C(F)F)no1)=O c1(-c2cccc(C3C(N4CCCC(c5cc(C)[nH]n5)C4)C3)c2)cccc(O)c1C N1(C(C2NC(=O)OCC2)=O)C2CCC1CN(C(=O)C(F)(F)c1nccs1)C2 C12(NC(COc3cn(C)nc3)=O)CCC(NC(=O)C(C)(O)C3CC3)(CC1)C2 N1(C(CC(=O)OCC)=O)CCN(C)CC1CNC(c1sc(C)cc1Br)=O C(C)(CSC)(C(=O)NC1(C)CCC(C)C1)NC(c1c(COC)cc[nH]1)=O N1(C(=O)Cc2cocn2)CC2CCN(C(c3ccsn3)=O)C2C1 C=C(C)CC(C(=O)NCC1(NC(=O)C2=C(Cl)CCC2)CCOCC1)OC C(=O)(CC(C(F)(F)F)NC(=O)Cc1ccc(O)cc1)N(CC(F)F)C(C)C c1(C(=O)NCC2CCC(NC(c3ccon3)=O)C2)cccnc1-c1ccncc1 N1(C(C2CC=C(C)CC2)=O)CCC(NC(c2cnc(C)cn2)=O)C(CO)CC1 c1(C(N(CC(CNC(c2cc(C)nn2C)=O)(C)C)C)=O)ccc2nccnc2n1 CC(C(=O)NCC1CN(CCN2CCCS2(=O)=O)CCCO1)C(F)(F)F C1(CNC(C2C(C=C)C2)=O)CCC(C)(C)CN1C(=O)CSc1ccc(F)cc1F c1(CNC(C(C)SC)=O)cccc(C(=O)N(C)Cc2cc(C)no2)n1 Cc1nn(C)c(C(=O)NCCCNC(C23CSC(C2)C3)=O)c1[N+](=O)[O-] N1(C(C2(O)CC2)=O)CCc2cc(-c3cc(F)ccc3[N+](=O)[O-])ccc2C1 C1(CC(N2CC(C(C(=O)NCC3CCC(=O)O3)OC)C2)=O)CCCC2CC12 Cc1cc(Br)ccc1-n1cc(CC(O)C(=O)NC2(CN(C)C)COC2)nn1 C1(CC(=O)NCCC(C)NC(c2cncc(C3CC3)c2)=O)OCCC1(C)C Cc1c(Cl)ccc2c1CN(CCC(=O)NC1CCCCCC1)CC2 c1(OC)ccc(CN2CC3CC2CN3C(c2csc(Br)c2)=O)c(F)c1F Cc1cnnc(O)c1C(=O)NCC(=C1CN(C(=O)Cc2ccc(Cl)cc2)C1)F C12(NC(C(C)CC#N)=O)CCC(CN(C(=O)Cn3cnc([N+](=O)[O-])n3)C1)C2 C(CC(=O)NC(c1ccccc1)C)(C(F)F)NC(CC(=O)OCC)=O c1(NS(CC)(=O)=O)ccc(C(=O)N(C(C)CNC(=O)CC2(COC)CC2)C)cn1 N1(C(C(C)N(C(C)=O)C)=O)C2CCC1CC(C(N1CCOCC1CCO)=O)C2 Cc1ccc(C(=O)NC2CN(C(C3CCS(=O)(=O)C3)=O)CCC2C)c(N=[N+]=[N-])c1 N1(C(CC(C)(O)CC(=O)O)=O)CCc2cccc(Br)c2C1.N12CC3CC3(C1)C2=O c1(C(CNC(=O)CC2CC2)NC(COCC(=C)C)=O)ccc(OC)cc1 c1(C(N2C(CNC(=O)CCOC3CCC3)COCC2)=O)cccc2cnccc12 N1(C(C(CC(C)C)NC(=O)OC)=O)CCC(C)N(C(=O)Cn2nnnc2C)CC1 N1(C(c2c(CCC)[nH]cc2)=O)CCC(C)(CC(=O)NCC(c2cn(C)cn2)O)C1 Cc1nc(NC(N2CCCCC2CO)=O)ccc1O C1(CC(=O)NC(CNC(CCc2cn(C)nc2)=O)C(C)(C)C)CCOC(C)(C)C1 C1(CCC)CN(C(c2ccc(F)c(SCC)c2)=O)CCN1C(=O)CCC1CC1 c1(OC(CC)C(N2CCC(C)(NC(=O)C3=C(Cl)CC3)C2)=O)ccc(C)cc1 C1(NC(C(F)=CC)=O)CCC(CNC(c2cc(-c3ccn(C)c3)[nH]n2)=O)CC1 C(=O)(C1SCc2cccnc21)N1CCCC(CNC(c2cc(N)nc(Cl)c2)=O)C1 c1(C(=O)NCCC(C)NC(c2cn(CCCC)nn2)=O)coc2c1C(O)CCC2 C(CCC(=O)N1CCC(CC(=O)NCCCc2cc[nH]n2)C1)SC C1(CNC(c2scc(C)c2)=O)CC2(CC2)CN1C(C1OCCN(C)C1=O)=O c1(C(C)C)cc(C(N2CCN(C(=O)C#CC3CC3)C(C(C)(C)C)C2)=O)ccc1O C(=O)(C#CC1CCCC1)N1CC(CN(C(Cn2nnc(C)n2)=O)C)OCC1 c1(C(N2CCN(C(C3(C4CCC4)CC3)=O)C3CC23)=O)cc2cccn2cn1 CCCCCC(F)C(=O)N1CCC=C(C(=O)NCC2(C)CC(C)C2)C1 C(CC(F)(F)C(F)F)n1cc(CNC(C2C(CC(N)=O)CCCC2)=O)nn1 C(=O)(CCC(F)(F)F)NCC(CC(=O)NCc1c(OC)nn(C)c1)OC C1(C)(OC)CCCN(C(c2cc(CNC(C3(CO)CCCCO3)=O)cs2)=O)CC1 C=CCC(CC(C)C)C(=O)NCC1CCC(NC(c2n[nH]c(C3CC3)n2)=O)C1 c1(CNC(C2(CNC(c3c(C)nn[nH]3)=O)CC2)=O)ccc([N+](=O)[O-])cc1 c1(CC(N2CC(S(=O)(=O)NC(=N)N)C2)=O)cnc2ccccc2c1 C1(CC(=O)O)CSCCN1C(=O)CCC(Cl)Cl c1(C(N2CCC(CNC(C(C3CC3)OC)=O)CC2)=O)c(C)[nH]c2ccc(Cl)cc12 c1(C(=O)NCC#CCNC(COCCC#C)=O)ccnn1CCC Cc1nc(CC(C)C)sc1C(=O)NC1(C)CCN(C(=O)Cn2cc(N)cn2)C1 C1(CC(N2CC(CCCCNC(c3c(C)ccs3)=O)C2)=O)CCCC(C#N)C1 C(=O)(C(C)(C)CC(C)(C)C)NC(CC(CC)C)C(=O)NC1CC(Cl)(Cl)C1 N1(C(Cc2ccc(C)s2)=O)C(CNC(=O)CC2CC(C)OC2C)CC2COCC12 c1(CC)nc(C(=O)NCC2(CNC(=O)C(C)=C3CC3)CC2(F)F)c(C)o1 c1(CC)nc(N2CCCC(NC(c3noc4c3COCC4)=O)C2)c(CC)c(Cl)n1 C1(C)(C(N2CCC(COCCOC)C2)=O)c2ccccc2CC1(C)C Cn1cc(CNC2CCC(F)(C(=O)O)C2)c2ccccc12 C#CCCCCCCC(=O)N(CC(=O)NC(CCC=C)C(=O)OC)CC c1(C(N2C(C)CC(NC(c3cc(OC)nn3C)=O)C2)=O)cccc2c1C(=O)NC2 CCCCCS(=O)(=O)CC(=O)NC1CCCC1NC(c1ccc2n[nH]cc2c1)=O C#Cc1ccc(C(N2CCCC2C(C)NC(=O)C=CC)=O)o1 C1(C)(C(=O)NCC(CC)NC(c2ccn3ccnc3c2)=O)Cc2ccccc2N1 c1(CN(CCCCC)CC(O)CC)ccc(OC)c(F)c1 c1(C(=O)NCC=CCNC(C2C(OC)CCC2)=O)cnc2onc(C(C)C)c2c1 C(=O)(C(C)CC(N)=O)N(CCCNC(CCC#CC)=O)Cc1cccnc1 CCCC(C(O)C(=O)NC1CC(=O)NC(=O)C1)NC(=O)CC1(O)CCCC1 c1(C(=O)NCC2N(C(Cc3n[nH]c(=N)s3)=O)CCC2)cnn2c1CC(F)(F)C2 N1(C(=O)Cc2ccc(F)c(Cl)c2)CCCN(C(C23CCCC2C3(F)F)=O)CC1 C1(NC(=O)COc2ccsc2)CCN(C(=O)CSc2ccccc2Cl)CC1 C1(NC(CCC(CC)C)=O)COC2(C1)CN(C(c1c(C)nc(O)nc1C)=O)C2 N1(C(C=C(CCC)C)=O)CCN(C)CC1CNC(=O)C(CO)OC C1(CNCC(c2scc(C)n2)C)CC12CCCCC2 C#CC1N(C(=O)C(C)(C)C(N)c2ccccc2)CC1(C)C c1(CCC(N2CC(C)C(CCNC(=O)C(C)(C)F)C2)=O)ccc2c(c1)CCO2 c1(-c2ccn(C)n2)ccc2ccc(C(=O)Nc3c(Cl)cc(C#N)cc3Cl)nc2c1 c1(C(=O)NCC2C(NC(C3(C(=O)OCC)CCC3)=O)CCC2)c(C)[nH]c(C)c1C C1(CC=C)(NC(CSCC=C)=O)CN(C(=O)CCCN2CCOCC2)C1 C(C(O)(COC)CO)NC(C(C)(N(C(C(C)OCC=C)=O)C)C1CC1)=O N1(C(C(=O)NC)COC(C)(C)C)CCc2c(ncn(C)c2=O)C1 C1(CC(=O)NCCCC(C)NC(=O)CC(C)(C)N(C)C)CCN(C)CC1 c1(CC)cnc(C(=O)NCC2CCN2C(c2ccc(CSC)o2)=O)nc1 C(c1cccc(Cl)c1Cl)=CC(N1C(CNC(c2cn(C)nn2)=O)CC1)=O C(=O)(C1CCc2ccc(Cl)nc21)N(CC(C)NC(=O)C(C(C)(C)C)NC(N)=O)C C1(CC(C)O)CCN(C(c2occc2CNC(=O)CCN(C)CCO)=O)CC1 CC(C)C(F)(F)CC(=O)NCC1CCCCC1NC(c1c[nH]c2ncccc12)=O Cc1nc(F)ccc1CC(N1CCC(Cn2cc(C(O)CC(C)C)nn2)C1)=O c1(OC)c(C)cc(C(=O)NC2CC2NC(C2CCC(=O)N2C)=O)cc1Cl c1(NC(=O)CC2CCCSC2)ccccc1.c12nc(co1)C(=O)NC2.C(CO)O C(CN1C(=O)OCc2ccccc21)NC(=O)Nc1c(C)cc(=O)n(C2CCSC2)c1 c1(C(=O)NC(C2CCN(C(C3(C(C)(C)OC)CC3)=O)C2)C)cc(C)cc(F)c1N N1(C(c2cc(SC)oc2)=O)CC2(C1)CN(C(c1sc(C)cc1C)=O)CC2CO c1(C(=O)NC2CN(C3=NCCS3)C2)cc2c(s1)CNCC2 N1(C(=O)C(C2CCOCC2)O)CCN(C(c2ccc(O)nc2)=O)CC(O)C1 C1(CN(C(=O)C(O)COC)CC)CCCN1C(c1cn(C)cn1)=O C(=O)(C#CC1CCCO1)N(C1CCN(C(CC2(C=C)CCC2)=O)C1)CC c1(C(=O)NCC2N(C(C(CC)n3nccc3C)=O)CC2)ccccc1O CCCCC(O)CC(=O)NC1(C(=O)N(CC(=O)OCCSC)C)CCCC1 C1(C(=O)NCC2N(C(c3cccc(=O)o3)=O)CCN(C)C2)CCc2nnnn2C1 c1(C(=O)NCC2C(NC(C3C(C)OC(=O)N3)=O)C2)cnc2ccccn12 C(CCC(=O)N1CCC(Oc2cccnc2)C1)NC(C(N(C)C)C1CC1)=O CN1CCCC(O)(CC(=O)NC2CCC(NC(=O)Cc3cccnc3)C2)C1 CC1CN(N2CCCC(CN(C)Cc3ccccc3)C2)Cc2cncn21 N1(C(C2(C(N)=O)CCC2)=O)CC=C(CCNC(=O)Cc2cc(C3CC3)no2)CC1 CCC(O)C(C)C(=O)NC1CCC(CNC(=O)CCC2CCC2)C1 c1(C(=O)NC(CCCC)CO)cccc(S(=O)(=O)N2CC3CC(F)CC3C2)c1 C(c1cc(F)c(O)c(F)c1)=CC(N1CC(CN(C(C(C)OC)=O)C)C2(C1)CC2)=O C(=O)(C(CCC(C)C)NC(C1CC(C)CC(=O)N1)=O)NCC(CC=C)(C)C CS(=O)(=O)c1ccc(NC(CNC(=O)CC(F)(F)F)Cc2ccccc2)nc1 c1(C(N2CCC(CC=C)(C(N3CCCC3CN(C)C)=O)C2)=O)cc(O)cc(=O)o1 C1(C)(C(N(C2CCCCN(c3ncc(Br)c(O)n3)C2)C)=O)CCCCC1(F)F C1(C(=O)NCCC(C(C)C)NC(c2cc(Cl)ccc2Cl)=O)CC1C1(C)CCCCC1 C1(CC(=O)NCCN2CCC(NC(C3CCO3)=O)CC2)CSc2ccccc2O1 c1(N2CCCC(NC(c3cnn(C(F)F)c3)=O)(CO)C2)c(Cl)cccc1[N+](=O)[O-] C1(NC(c2c(SC)cnn2C)=O)CS(=O)(=O)CC1NC(c1cc(C)nc(O)c1)=O n1(N)ncc(C)c1COSCC(CO)OC.C(=O)(N)OC C(=O)(C(C)(COCC)CC)NC1C(N2CCN(C(CCC)=O)CC2)COC1 C(=O)(CCC(=O)N1CCCCC1C1CCCN(C(=O)CCc2cnn[nH]2)C1)NC C=C(C)CC(C(=O)N1CC2CC2(CNC(C2CC23CCCC3)=O)C1)NC(C)=O C1(O)(CCNC(c2c(C)nc(N(C)C)s2)=O)CCN(C(C2CSCCS2)=O)CC1 C1(C)(NC(=O)NCCCc2ccc(OCC)c(OC)c2)CCC(=O)N(C)C1 Cc1cc(C(=O)NC2CC(CNC(=O)C(c3cccnc3)O)CC2O)nc(O)c1 C1(C(=O)Nc2cccc(C)n2)CC2CC1CN2C(c1cc(C#N)c[nH]1)=O C(CC(=O)NCc1cccc(NC(C2CC=CCO2)=O)c1)(C(F)(F)F)OC N1(C(C(CCC)C)=O)CCOCC(C)(CNC(=O)CCc2ccc(CC)cc2)C1 N1(C(C(CSC)(C)C)=O)CCC(NC(C2CCN(c3ccncc3)C2)=O)C(O)C1 C1(C)(C(N2C(CCC(C)C)CCC2)=O)CCCN(C(c2cccc(=O)o2)=O)C1 C(C(=O)C(C)N1CCC1(C)c1ccccc1)OCCOC c1(NC(c2ccc(-c3cc(C)cc(F)c3)cn2)=O)ccc(Br)c(Cl)c1C Cc1ccc(NC(C)C)c(C(N2CC(NC(=O)CCC3CC3)CC(F)C2)=O)c1 N1(C(=O)Cc2nccs2)CC(CO)C2(C1)CN(C(c1n[nH]cc1Cl)=O)C2 c1(C(=O)NCC(C2CC2)NC(C2CC(F)(F)C2)=O)ccc2nc(C3CC3)oc2c1 c1(-n2ccc(C(N3C(C=C)CC3)=O)n2)cc(F)cc(F)c1.C12CCN(CC1)C2 C(C(O)C(F)(F)C(F)(F)F)NC(=O)NC(C(=O)OC)C(C)(F)F C(CC1=CCN(C(=O)CC2(O)CCCOC2)CC1)NC(c1cc(Cl)nnc1Cl)=O N1(C(CC(CC)C2CC2)=O)CCCCC2(CCN(C(c3cnnc(O)c3)=O)C2)C1 CN=c1ccc(C(N2CCCC(CCNC(=O)C=Cc3cccs3)C2)=O)c[nH]1 N1(C(C(C)OCC)=O)C(CNC(=O)C=Cc2ccc(F)c(Cl)c2)CC2CCCC12 C=C(C)CCC(c1nnnn1CCOC)NCc1nc(CCc2ccco2)no1 c1(C(=O)NC2C(NC(C(c3ccc(Cl)cc3)OC)=O)C2)ccc2ccsc2c1 C1(CNC(CCC2(C)CC2)=O)CCN(C(c2c[nH]nc2Cc2ccccc2)=O)C1 C1(F)(C(N(C2CCN(C(c3ccnn3CC(F)F)=O)C2)C)=O)CCCCC1 C1(C(=O)NCC(C)N(C)C(=O)OC(C)(C)C)COCCC1(F)F C1(C(=O)NC2CCC(F)CC2)(CC)CCN(C(c2ccc(Cl)o2)=O)C1 C#Cc1cccc(C(=O)NCCC2CCCN(C(=O)CC(CC)SC)C2)c1F c1(C(=O)NC(CN(C(C2(N(C)CC)CCCC2)=O)CC)C)cc(C)n(C)n1 C(C(=O)Nc1ccc(F)cc1)(C1=NOC2(CCC2)C1)N1CCCC(C)(CC)CC1 C1(NC(=O)CC23CCCC2C3)CCCCN(C(=O)Cn2ccc(O)nc2=O)C1 S(=O)(=O)(c1ccc(=NCc2cccnc2F)[nH]c1)NCC1C(C)(C)C1 C1(NC(Cc2ccc(C)o2)=O)CCCCCN(C(C2CCCCCS2(=O)=O)=O)C1 C(=O)(CCC(C)(C)C(=O)OC(C)(C)C)N1C(CNC(C2(CC)CCC2)=O)CCC1 CON(CCC(=O)NC1CCOCC1C)C(=O)CNC(N)=O N1(C(C2N(C)CCOC2)=O)C2CCC1CN(C(C1(OC(C)C)CCC1)=O)C2 C12(NC(C#CCNC(C3C(C)CCC3)=O)=O)CCC(O)(CC1)CC2 C(CC(F)F)(C(=O)NCC1(F)CCN(C)C1)N(C(C(CCOC)C)=O)C C1(C(N(CCC#N)Cc2ccccc2)=O)C2CN(S(=O)(=O)C(Cl)(Cl)Cl)CC12 c1(C(N2CC(C)C(CCNC(=O)CN(C)CCO)C2)=O)cc(S(N)(=O)=O)co1 c1(C(=O)NCC2CCCC(NC(C3(C)CC=CC3)=O)C2)cc2ccccc2o1 N1(C(CC(C)CC(F)(F)F)=O)CCC(O)(C2(NC(c3cnn[nH]3)=O)CC2)CC1 C1(CC=C)(NC(=O)C=Cc2ccncn2)CCCN(C(C2CCC(=O)NC2)=O)C1 C(=O)(CC(C)(C)CC(F)F)NCC1CC(NC(C(C)OCC=C)=O)C1 N1(C(C(C2CC(F)(F)C2)OCC)=O)CCCC(C)(NC(=O)C(=O)NCC(F)F)C1 C1(CNC(C(N2CCCC(C)(C(F)(F)F)C2)=O)=O)CCCC2CCCN12 CCCCCCC(=O)N(C1CCCC1)CCNC(c1cccc(OC)c1)=O C1(C)(CNC(C=C(C)C)=O)CN(C(=O)CC2CC3(CCCC3)CO2)C(C)(C)C1 c1(CN2CC(C(=O)Nc3cccc(Br)c3O)C(O)CC2)ccc(Br)cc1[N+](=O)[O-] C=CCCCC(C(=O)N(C(CO)C(C)C)C)NC(C1CC1(Cl)Cl)=O CCC1=NOC(CC(=O)NCCCC(=O)NCCc2ccnc(C)c2)C1 Cc1cc(O)ccc1C(=O)NC1CC(CCNC(=O)Cn2cc(C(F)F)cn2)C1 C1(O)(CCNC(c2cc(C(C)C)on2)=O)CCN(C(C2CC=CCO2)=O)C1 C(CC(C)C)C(=O)N1CCC(C(=O)NOCC=C(C)C)C12CC2.CC(C)CCC=O C(=O)(CCS(N)(=O)=O)OCC1N(C(=O)OC(C)(C)C)C(C(F)(F)F)C1 C1(C(=O)OCC)CN(C(c2c(OC)ccc(F)c2OC)=O)CC(F)(F)C1 C(=O)(C1CCc2ccccc21)N1CC(CCC)N(C(c2cc(C)oc2C)=O)CC1 C1(N(C(C(N2CCC(C)C2)=O)=O)C)CN(C(=O)Cc2c(Cl)cnn2C)CCC1C C1(C)(CNC(C2N=C(C)SC2)=O)CCCN1C(c1cc(CC2CCC2)c[nH]1)=O C1(CNC(c2cc(C3CC3)ccn2)=O)CCC2(CCC3(CC2)OCCO3)O1 Cc1cc(C(=O)NCC2(C(N)=O)CN(C(c3cnn(C)c3C)=O)C2)sc1C N1(C(c2cc(CC)n(C)n2)=O)CCC(Nc2ncccn2)C(O)C1 CCC(C)C(C)C(=O)NC(C1CCCCC1)CC c1(SC)nc(N2CCC(NC(c3ccc(Br)cc3Br)=O)CC2)ncc1F C(=O)(C(C)CCOC)N(CCCNC(c1cccc(=O)o1)=O)CC c1(OCC)ccc(NC(=O)NCC2(Nc3ncccc3F)CN(C)C2)cc1 C=CCC(CNC(=O)Cc1ccc(C)cc1)C(=O)NCc1cn(C)nn1 C1(C(=O)NCC2CCC(F)C2)CC2CC2N1C(=O)Cc1cccc(O)c1 c1(C(=O)NCCCN(C(C)C)C(c2ccncc2Br)=O)cc(O)cc(F)c1 CC1CN(C(C2CC3CCC2N3C(=O)C(=O)NCC(C)(C)C)=O)CCC1(F)F c1(C(=O)NC2CCN(C(CCCCOC)=O)CC2CO)nc(Cl)cc(N)c1Cl c1(C(N2CC(OC)C(NC(C3Cc4nccn4C3)=O)C2)=O)cc2ccccc2o1 n1(CC)c(Sc2ccc(Br)c(F)c2)nc2ccc([N+](=O)[O-])cc2c1=O c1(C(N2CCCC(N(C(C)C)C)C2)C(=O)NCCC2CC2)nc2c(s1)CCCCC2 c1(C(=O)NC2C(CNC(CNC(=O)OC)=O)CCC2)cccc2c1C(F)(F)CC2 N1(C(CC#N)=O)CCC(NC(c2ncccc2C(F)(F)F)=O)C(F)C1 C1(C(N2CC(NC(C(CC)(C)C)=O)C(C)C2)=O)CN2CCC1CC2 C(=O)(C(F)CC(C)C)N1CC(NC(c2cn(CCOC)nc2C)=O)C(OC)C1 C1(N(C(C2CN(C)C(=O)C2)=O)C)CN(C(c2csc3nccn23)=O)CC12CC2 c1(C(N2CCC(C)(NC(c3cc(C)c(C)nc3)=O)C2)=O)nccc2occc12 Cc1cc(-n2nnnc2C2(Nc3cccc(Cl)c3C)CCN(C)C2C)ccc1F C=CC(C)(O)C(=O)N1CCN(CCN(C(=O)CC(=C)Br)C)CC1 N1(C(c2ccc(CC)[nH]2)=O)CC(O)CCC1C(=O)NCc1nc(CO)n[nH]1 c1(C(N(C(CNC(c2nncc(OC)c2)=O)C2CC2)C)=O)ncnc2ccsc12 C1(C(=O)NCCC(C)NC(=O)CCCc2cccc(Cl)n2)CC2(CCC2)CO1 N1(C(CCc2n(C)ncc2)=O)CC2CCCC(C1)N2C(=O)C1=CCCOC1 N1(C(CSCc2ccc(C)cc2)=O)C2CCC1CC(NC(C1CC(=O)N1)=O)C2 O=C1CC2(C(N3CCC(C(=O)O)CC3)=O)CNCC2N1 c1(C(=O)OC)ccc(=NCC2CC(C)N(C(=O)CC3CCOCC3)C2)[nH]c1OC C1(NC(C(CSC)OC)=O)CC(O)CN(C(=O)CC2(C)CC2)C1 N1(C(C2N(C(c3ccc(NC)cn3)=O)CC(=O)NC2)=O)CCc2nc(C)[nH]c2C1 c1(CS(N2CCCC2CC(c2ccco2)O)(=O)=O)cc(I)c(F)cc1F CCCC(C(=O)N(C)C)NC(=O)CCC(C)NC(C1CC(=O)CS1)=O C(C)(C(=O)NOCCF)N(C(c1ccncc1)=O)CC C12(CNC(C(n3cnc(C#N)n3)CC)=O)CC(NC(c3ccsc3C)=O)(CO1)C2 N1(C(CCOCCOC)=O)CCCC(CC)C1C(=O)NCC1(C)CCCO1 CN1CC(=O)N(CC(=O)NCC2CCCC(NC(=O)Cn3nccn3)C2)C1=O Cc1ccc(SCC(N2CCC(C(C)NC(=O)COCCCF)C2)=O)cc1C C1(N(C2CCCNC2=O)C(CC)(COC)c2nnnn2C)COCCC1O N1(C(Cc2cc(C)on2)=O)CCC2(CNC(C3CC34CC4)=O)CCCC12 c1(C(=O)NCC(c2cc(C)oc2C)(C)O)cc([N+](=O)[O-])ccc1O CC(N(C)N1CCCC2(CC1)CC2(F)F)c1ccc(-c2ccc(Cl)cc2)o1 CCC(C)(F)C(=O)NCCC(C)NC(=O)C(O)CC1CN(C(=O)OC(C)(C)C)C1 N1(C(C(C)OC)=O)CCOC2(CCN(C(c3noc(C)c3[N+](=O)[O-])=O)CC2)C1 C(CCCCC(=O)N1CC(CCNC(=O)CSc2nnnn2C)(OC)C1)OC c1(CCC)ccc(C(=O)NC2COCC2NC(C2CCOC2C(F)(F)F)=O)s1 c1(CC)nc(C(=O)N(CC(=O)NC(C2CCN(C)C2)C)C(C)C)co1 N1(c2nc(Cl)nc(C)n2)CC=C(CCNC(C2CCCCS2)=O)CC1 c1(C2(C(=O)NC(=O)CC3(CO)CC3)CC2)ccc(C)nc1.C12(CNC(=O)C1)NC2 C1(C(CNC(C2NCCCC2C(F)(F)F)C)C)CCC(F)(F)CC1 N1(C(C(CC=C)CC)=O)CCC2(CC2)CC1C(N1CC(OC)CC(C)C1)=O c1(NC(C2(C)CCCN2C(=O)C(N)=O)=O)ccc(Cl)c(I)c1 CCC(C)(CNC(=O)C(CNC(C1CCS1(=O)=O)=O)OC)C(N)=O C(=O)(CC1C(=O)Nc2ccc(F)cc21)N(C1CN(C(C(C(CC)C)OC)=O)C1)C Cc1nn(C)c(Cl)c1C(N1CC2(CNC(=O)CC3C=NN(C)C3=O)CCC1C2)=O C(C1=NOC2CN(C(=O)C#CC3CCOCC3)CC12)NC(c1cscn1)=O N1(C(CCCOC(C(C)C)=O)=O)CCC(C(CO)NC(=O)CC2(CO)CC2)CC1 O=C1CCN(C(C23CC2CN(C(C2COCOC2)=O)C3)=O)CCN1 c1(C(N2CCCC(N(C(C3CC(F)(F)C3)=O)CC)C2)=O)c(N)cc(Cl)nc1Cl c1(C(=O)NC2CCCN(c3c(OC)cccc3)C2=O)ccc(S(N)(=O)=O)cn1 C1(NC(CCCOCC)=O)Cc2ccccc2C1NC(c1cc(Cl)ccc1Cl)=O C1(C(=O)NC2(CC=CC(=O)NCCc3onc(C)n3)CCC2)C2CC3C(C2=O)C13 N1(C(CCCN(C(C)C)C)=O)CC2CC(C1)N(C(=O)C=CSc1ccccc1)C2 CC1(CNC(C2CCNC(=O)C2)=O)CCCN1C(=O)CC1C=CS(=O)(=O)C1 C(=O)(CC(C(F)F)NC(c1cccc(CO)c1)=O)Nc1ccc(CC)cc1 N1(C(c2c(C)csc2)=O)CCOC(c2ccnc(N3CCCCC3)n2)C1 N1(C(CCCC#C)C(=O)NC2(C)CC2)CCc2c(F)cccc21 CC(C)C(C(=O)NC(C)CNC(=O)C(C(C)C)N(C)C)n1cncn1 C1(O)(CN(C)C(C2CCCCN2S(C)(=O)=O)=O)CCN(C(=O)C=CC2CCC2)C1 C1(NC(Cn2ccc(C)n2)=O)CC2C(NC(C3CC(C)(O)C3)=O)C2C1 C1(CNC(C(C)N2CCCC2)=O)N(C(=O)COc2ccsn2)CCCC1(C)C C1(NC(c2n(CC)ccn2)=O)(CNC(=O)CC(O)C2CCCC2)CCCCCC1 n1(CC(=O)NCC2C(CNC(c3nc(C)nn3C)=O)C2)cc(Cl)c(O)nc1=O c1(N(CCS(N)(=O)=O)C)nccc(=NCCCc2ccc(CO)cc2)[nH]1 c1(CCCSCC)nc(C(c2cn(C)nc2C)C2CCC2)n(-c2ccc(F)nc2)n1 c1(NC(=O)NCC(=O)C2CC2c2ccno2)ccccc1Br N1(C(C2(CSC)CCC2)=O)CC2CC2(CNC(c2csc(-c3ccoc3)n2)=O)C1 c1(C(N2CCCCC2c2cccs2)C(=O)NC2COC2)nnc2n1CCC2 CN1CCN(C(=O)CCCNS(C)(=O)=O)CC1CNC(C1COC(C)(C)C1)=O n1(CC)ccc(C(=O)NC2CCC(C)(NC(c3cnc(OC)s3)=O)CC2)cc1=O N1(C(c2n(C(CC)CC)ncc2)=O)CCCCC(NC(C2CNC(=O)C2)=O)C1 Cc1cc(C(N2CCC(NC(C3CCCN3N=O)=O)C2)=O)ccc1[N+](=O)[O-] Cc1cnc2ccc(C(N3CC(O)CC3(C)C(=O)O)=O)cn12 N1(C(C(CC)O)=O)CC2CC1C2C(=O)NCC(C)(O)CCO Cc1ccc(CN2CCC(O)(CC(N3Cc4ncsc4C3)=O)CC2)c(Cl)c1 CCC(CC(F)(F)F)C(=O)NC(C)(CNC(=O)Cc1cccnc1C)CSC c1(SC)cnn(C)c1C(N1CC(NC(C2CCCC2C(F)F)=O)C(O)C1)=O c1(CN2CC3(N(C(c4cc5cccnn5n4)=O)CC3)C2)ccc(F)c2ccoc12 C(C(C)(C)C(=O)NC(C)CCCCNC(=O)CC1CCCC1)SC c1(CC(=O)NCC(C)N(C)C(c2cc(C(=O)C(F)(F)F)c[nH]2)=O)nnc(S)n1C C(=O)(CC(CC)C(C)(C)C)NCC(CCC)NC(C=CCCC)=O c1(C(=O)NCC(N(C(CC2CN(C)C2)=O)C)C2CC2)ccc2oc(=O)oc2c1 C#CCC(C)(C(=O)N1CCNC(=O)CC1)NC(=O)Cc1ccsc1 C1(CN(C)C(C2(O)CCSC2)=O)C2CN(C(=O)CC3CSC3)CC12 C1(C2CC2)(CNC(C(c2cncnc2)C)=O)CCN(C(=O)C=C2CCCCC2)C1 S(=O)(=O)(c1cc(CC)cc(C)n1)N1C(CC#C)CCCC1 CP(C)(=O)C1CCC(Nc2cc(F)cc(F)c2)C1 c1(OC)nc(N2CCC2C(=O)Nc2c(Br)cnn2C)nc2[nH]cnc12 N1(C(c2[nH]cc(CC(C)C)c2)=O)CC(F)(F)CC1CNC(=O)CC1CCCCC1 c1(OC)cccc(OC(C2CN(C(=O)SC)C2)=O)c1.C1CCN1CCC#N C(=O)(NN1CCN(Cc2ccccc2)CC1)c1c(Cc2cn(C)nc2)ccs1 C=C1CC2(C1)CC(C(=O)NCC(CC(C)C)NC(C1(O)CC1(C)C)=O)C2 C1(C(N2CCOCC(NC(c3noc(CC)c3C)=O)C2)=O)CN2CCCC2CO1 C1(C(NOC(CCC)C2CC2)=O)(NC(c2cnn(C(F)F)c2)=O)CCSC1 C(=O)(CC1NC(=O)c2ccccc21)NCC1C2CN(C(C3CC(SC)C3)=O)C1C2 C1(CC)CCCCC1OCC(N1CC(C(N)=O)(CNC(C2CCCO2)=O)C1)=O Nc1cccc(C(F)F)c1C(=O)NCC1(O)CCC12CCC2 c1(NC(C(c2ccccc2)OC(C)=O)=O)cc(C(=O)N(CCO)CCO)n(C)c1 Cc1ccc(C(F)(F)C(=O)NCC(C2CC2)N(C)C(C2(CN(C)C)CC2)=O)nc1 c1(C(=O)NC(C(=O)OCC)CCc2ccccc2)cc([N+](=O)[O-])cc(Br)c1F Cc1ccnc(NC(C2COCCN2C(c2cnc(O)nc2O)=O)=O)c1C c1(C(=O)NCCCN(C(=O)C=C(C)C(F)F)CC)[nH]c(C)c(C(C)=O)c1C c1(C(=O)NCC(c2ccc(NC)cc2)N(C)C)cc2[nH]c(=O)cc(C)n2n1 C=CCC(C(=O)N1CCC(N(C(=O)CCC(=O)n2cc(Br)cn2)C)C1)OC CC1CC(CNC(=O)Cn2cccn2)CN1C(=O)C(C)CSc1ccc(F)cc1 Cc1ccc(C(N2CC(NC(c3onc4ccccc34)=O)C(C)C2)=O)c(F)c1F Cc1cccc(C(=O)NC2CCC(C)(CNC(=O)CCCc3ccsc3)C2)c1 n1(CCC(C)=O)cc(CNC(C2(CC(C3CCOC3C(C)C)=O)CC2)=O)nn1 C1(C(=O)NC2C(NC(c3ccco3)=O)CCC2)CCC(F)(F)C1 C(=O)(CS(=O)(=O)C(C)C)NC1C(OC)CN(C(C2CCOC(=O)N2)=O)C1 CC#CCCC(=O)NC1(CC=C)CCN(C(C2CCC(F)(F)C2)=O)C1 CCCCC(CC)CC(=O)N1CC2CCC1(CNC(c1ccnnc1O)=O)CC2 CCCCCC(C)CC(=O)NCCC1(CNC(c2c(C)nc(=N)[nH]c2C)=O)CC1 C1(CC(=O)NC2CCCC(NC(=O)COCC(F)F)C2)(COC)CCOCC1 c1(C(=O)NC2(CN(C)C(C3CC(=O)N(O)C3)=O)CC2)ccc(C2(C)CC2)cc1 C1(C(=O)NCC(CN(C(c2cnc(C)o2)=O)C)C)C2CCCCC12 c1(CCC(=O)NCCCOCCNC(=O)CCC=CBr)ccc(Cl)cc1 C1(C(=O)NCCNC(C2C3CCC2(c2cccnc2)C3)=O)CCC2C1C2(F)F N1(C(Cc2cc(C)no2)=O)CCN(C(c2ccc3c(c2)CCC3)=O)CC1C#N C1(C)(COCC)CCN(C(=O)C(=O)Nc2cccc(-c3ccc(Br)cc3)c2)CC1 c1(C(=O)NCC2N(C(CCC(CC)OC)=O)CC=C2)cc2sc(Cl)cc2[nH]1 C(c1cccc(O)c1)=CC(=O)NCC1CCCN(C(C2(C=C)CC2)=O)C1 CCC(C(=O)NC1(C(=O)NCC2(C3(O)CCC3)CC2)CC1)C(=O)c1ccc(Cl)cc1 Cc1ccc(F)c(C(=O)NCCCN(C(=O)C(N2CCCCCC2)C)C2CC2)c1 C(C(C)(C(=O)NCCN1CC(CF)C1)NC(=O)CC1CCOC1=O)SC c1(NC(C2CCC=CO2)(c2nnnn2C2CCCCCC2)C)cnn2c1OCCC2 N1(C(c2ncn(CC)n2)=O)CCC(C(F)(F)F)C(NC(=O)C2=NOCC2)C1 N1(C(C)C)CC(CNC(C2(C(=O)N)CC2)=O)C1.C12(CC1)OC2.N(C)C C1(C(N(C2(c3onc(C)n3)CC2)CC(=O)NC2(C#N)CCCO2)=O)CCN(C)C1=O C1(CN(CC(CCC=C)O)C)CCOCC12CCC2 CCC(C(=O)NC1CCC1NC(c1sccc1Br)=O)C(C)C c1(C(=O)NCC(=C)CCNC(=O)CC(CC)C2CC2)nccc2ccsc12 CCCC(=O)NCC(=O)NCC1(C(C)NC(=O)CN(C)C)CC1 C(C(CC(C)C)C(=O)N1CCNC(=O)C12CC2)NC(c1c(C)oc(C#N)c1)=O c1(C(=O)NC2C(CC)N(C(=O)CCS(=O)(=O)CC)CC2)cc(F)cc2ccoc12 C1(C(=O)NCC(C)OC(F)F)CCC(C)(C)N(C(=O)CC2(O)CCOCC2)C1 c1(OCC#C)ncccc1C(=O)NC1CN(C(C2CSCN2C)=O)CC1C CC(C)CCC(=O)NCC1(C)CCC(NCc2coc(Cc3ccccc3)n2)C1 C(Cc1ccccc1)(CCNC(c1scnc1Cl)=O)NC(=O)CCc1cnn[nH]1 C(=O)(C(CC)(CC)OC)NCC(C(=O)NCc1cn(CC#C)nc1)OC C(=O)(CC(F)(F)C(F)F)N1CCC(CNC(c2ccn(C)c2)=O)C1 c1(C(N(CCC(C)NC(C2(C)CC(=C)C2)=O)C)=O)cccc(N)c1O C1(NC(C2CC(=C)C2)=O)CC2(C(=O)NC3CC3C3CCC3)COC1C2 N1(Cc2ncn(C)c2)CCC2CN(C(c3ccnc(N(C)C)c3)=O)CC2C1 c1(N2CCC(CCNC(=O)C(c3ccccc3)C3CC3)C2)ccccc1[N+](=O)[O-] c1(-c2c(C)cc(F)nc2)n[nH]c2cc(C(=O)Nc3nccs3)ccc12 c1(OC)ccc(CC(N2CCCC(c3nc(C)c(C(=O)O)[nH]3)C2)=O)cc1 C(=O)(C(C)CN(C(=O)COCCc1cccs1)C)NC1(CC(=O)OC)CC1 O=S1(=O)CCC2CCN(C(=NCc3cccs3)NC3CN(C4COC4)C3)CC2C1 c1(C(=O)NC2CN(C(c3ccc(OC)c(Cl)c3)=O)C2)sc2ccccc2c1Cl N1(C(C(Br)=C(C)C)=O)CCC(c2cc(CNC(c3ccc(C)o3)=O)on2)CC1 CC1CN(C(C2CC3(C2)CC3(F)F)=O)CCC1N(C(=O)C(=O)NC1CC1)C Cc1cc(C(=O)NC2CCCCCN(C(=O)C(C)n3cccn3)C2)cc(C)c1O c1(C2(C(=O)NCC3CCN(C(COCC(C)C)=O)C3)CC2)cccc(F)c1 Cn1cc2c(n1)CCCC2C(=O)N1CCC(NC(c2ccc(Br)o2)=O)CC1 CC(C)C(CCN(C)C(C1(Br)CC1)=O)NC(c1cccc(O)c1)=O N1(C(C(C(CC)C)O)=O)CC(C)CN(C(c2cnn(C3CC3)c2)=O)C(C)C1 C1(CNC(c2nn[nH]c2C(F)(F)F)=O)CC2(CCN(C(=O)CC3CCC3)C2)CO1 C12(C(=O)NCC3(NC(C(CC)n4cncn4)=O)CC3)CC3CC(CC(C3)O1)C2 C1(C(N2CCCC(CCNC(C=C(COC)C)=O)C2)=O)CCc2n[nH]cc2C1 C(=O)(CCC(CF)CF)NC1C(NC(c2c(C)cccn2)=O)C1 c1(COC)ccccc1C(=O)NC(CCN(C)C(C1CCN1C)=O)C(C)C C#CCC(C(=O)NCC1(CNC(C2CCC(C(N)=O)CC2)=O)CC1)C1CC1 C1(C(N(C(C)CNC(=O)CSc2nnnn2C2CC2)C)=O)C2CCCCC12 c1(OCC)ccc(C(=O)CCC(=O)N2CCC(N(C)C(C3CCSC3)=O)C2)cc1 C1(NC(=O)CCC2CCCO2)CC(F)(F)CC1NC(c1ccco1)=O N1(C(c2cc(C)ncc2)=O)CCCC(C)(CNC(=O)Cc2ccc(Br)s2)C1 CC1CCC(Cl)=C(C(=O)NC2CC2CNC(c2cc(-c3ccncc3)on2)=O)C1 c1(C(N(C2CCCN(C(c3cccnc3CO)=O)CC2)C)=O)cc(O)cc(=O)o1 C1(NC(c2ccc(NCC3CC3)nc2)=O)CCN(C(c2ccc(O)cc2)=O)CC1 CCCC(C(=O)NCCN(CCOc1ccccc1)CC)OCC.C1CCCC1 N1(C(C(COC)NC(C)=O)=O)CCCC2(C1)CN(C(=O)CC(=O)NC)C2 N1(C(C(C)(F)F)=O)CCC2(CCCC2NC(=O)CSCc2ccccn2)CC1 N1(C(c2c(C)cccc2Cl)=O)CCC2C(C1)CN2C(C1C2COCC12)=O O=C(C1c2c[nH]nc2CN1C(=O)CC1CSC1)NCCF N1(C(C)C)CCCCC1C(=O)NCC1C=CCN(C(=O)CC2CC(F)(F)C2)C1 C12(C(=O)NC34C(CN(C(c5cccc(CCC)c5)=O)C3)C4)CCCC(CO1)C2 N1(C(c2cc3n(n2)CCC3)=O)CC2CCC2(CC(N2C3CCC2CC3)=O)C1 N1(C(COCC(C)C)=O)Cc2ccccc2C(NC(C23CC(C#N)(C2)C3)=O)C1 c1(C(CNC(C(CCC)OC)=O)NC(=O)CC(C)(C)O)ccc(F)cc1F c1(C(=O)NCC(CNC(CC(C)(C)SC)=O)F)cccc(Cl)c1[N+](=O)[O-] CC(C)(Cc1cn(CC2CCN(C(=O)CCCn3ccnc3)C2)nn1)CO c1(C(=O)NC(C(C)NC(CN2CCC(C)CC2)=O)C)cc(S(N)(=O)=O)cs1 Cc1nc(S(=O)(=O)Oc2ccccc2)cn1C.c12cc(C)c(o1)c(=O)o2 N1(C(CC2C(C)=NNC2=O)=O)CC(C(=O)NC2CCNC(=O)C2)C(C)(C)C1 C=C(C)C1CN(C(=O)CCC(CC)NC(=O)C(C)(C)F)CCO1 C(=O)(CC(O)C(C)C)N(CC)CC1CCCN1C(c1ccncc1O)=O CC(=O)CCCCC(=O)N1CCCCC2CC12 C1(NC(CSC)=O)CCC(N2CCN(C(=O)C=Cc3sccc3C)CC2)CC1 c1(OC)c(F)ccc(C(N2CC3CC2CN3C(=O)CC2CCC(=O)N2)=O)c1F N1(C(c2cc(Cl)c(Br)cn2)C(=O)NCCN2CCOCC2)CCc2c(Cl)cccc21 N1(C(c2cc(F)cc(F)c2O)=O)CCc2c(C(N3CCC(F)C3)=O)csc2C1 C1(NC(c2cccs2)=O)CN(C(=O)C=CC2CCCC2)CC1C1CC1 C(=O)(CP(C)(C)=O)NC1(C2N(C(CNC(c3ccn(C)n3)=O)=O)CCC2)CC1 c1(C(=O)NCCCN(C)C(C2(CF)CC2)=O)ccc(O)nc1Cl N1(C(CCC=C)C)CCC2(CC1)CC2C(N1CCC(N2CCCC2)CC1)=O N1(C(C#CC2(C)CC2)=O)CC(NC(c2cc(=O)cc[nH]2)=O)C2CCCCC12 c1(NC(C(C)NC(C(CC)n2ccnc2)=O)=O)c(C)n[nH]c1C C1(C)(CNC(C2(CC=C)CC=CC2)=O)CCCN1C(C1CCC(C(N)=O)CC1)=O Cc1c(F)ccc(Cl)c1C(=O)NCC1(CNC(C2CCC2)=O)CCOCC1 C1(N(C(C(C)c2ncco2)=O)C)CCN(C(C2CCC2C(F)F)=O)CC1 C1(CCC)COCCN1C(=O)C(C1CCC1)NC(=O)C(C)=C1CC1 C(=O)(C1CCc2ccc(Cl)nc21)N1CCC2(CC(CNC(CCOC)=O)OC2)C1 N1(C(C(CC#C)(C)C)=O)CC23CCCC2(C1)CN(C(C1CCN(OC)CC1)=O)C3 C1(NC(COCCC)=O)CCCN(C(c2nn(C)cc2Br)=O)C1 c1(CCC(=O)N(C(CCC)=O)CC(C)NC(C)=O)c(C)noc1C C1(C(=O)NC2CC(N(C(C(C)OCOC)=O)C)C2)C2C3CCC(C3)C12 N1(C(Cc2c(OC)ccc(C(F)(F)F)c2)=O)CC(C2CCC2)C1C(=O)OC C1(NC(c2ccc(Br)c(CO)c2)=O)CCN(C(=O)C(=O)C2CC2)CC1F c1(C(=O)NCCC2CCCN(C(C3CCCSS3)=O)C2)cccc2ccncc12 C1(C(=O)N(C(C)C)CC)CCN(C(=NCC2CC2)NCc2ncnn2C)CC1 c1(C(=O)NC2CCC(NC(CC3C(OC)CC3)=O)C2)ccc(OC(C)(C)C)cc1 c1(C(=O)NCCCC(C)NC(CCc2cnc(C)o2)=O)cccc(Cl)c1O c1(C(=O)NC2CCC(CCNC(C(C)=CC)=O)C2)cnn2c(OC)cccc12 c1(C(N2CCC(C)C(NC(c3cccc(F)c3F)=O)C2)=O)n[nH]c2c1CCOC2 C1(C)(CNCc2cccc(OCCOC)c2)CCC(=O)NC1 C1(COCC)NCCC1C1CC1.C1C(C)(C)C(=O)N1 C1(C)(CC)CC(NC(=O)CC(C)(C)COC)CN1C(c1ccc(Cl)s1)=O CC(C)(F)CCC(=O)NC1CN(C(C2CC(F)(CF)C2)=O)CCC1CO C1(NC(C2CCN2C(=O)C(c2ccccc2)O)=O)CC2(C1)CC21CCC1 C1(C2CN(C(C3CCC3c3ccccc3Cl)=O)C2)(NC(c2scc(C)c2)=O)CC1 C1(NC(CS(C)(=O)=O)=O)CCCCCCC1NC(=O)CCC1CC1 c1(CC)ncoc1C(=O)NCCCCN(C(=O)CC1(CN(C)C)CCCC1)C C(=O)(C(C(C)O)N(C)C)NC1CC(CCNC(c2cc(CC)on2)=O)C1 c1(C(=O)NCC(C)N(C(=O)Cc2cnns2)C)cc(Cl)c(O)c(Cl)c1 N1(C(c2c(CC)cco2)=O)CC2CCC(C1)N2C(C12CC(C#N)(C1)C2)=O C#CCC(C)(C(=O)NCCNC(=O)N(C)C)NC(C1CC1C(=O)OC)=O C(=O)(C1=Cc2ccccc2C1)N(CCC(C)NC(C1CC(CC2CC2)C1)=O)C c1(C(C(=O)N(C2CCOC2)CC(=O)OCC)(F)F)ccc(OC)c([N+](=O)[O-])c1 N1(C(C(C(=C)C)(C)O)=O)CCCC2(CCCN2C(c2ccn3cnnc3c2)=O)C1 Cc1ncc(CN2CC(F)CC2C(=O)NCCN2CCCCC2C)cn1 C1(C(=O)NC(c2nc(C(=O)NCc3cc(O)ns3)co2)C)OCC2CCCC12 c1(C(c2nnnn2C2CCOC2)NCCOCC(=C)C)cc(CC)no1 CC(C)CC(C(=O)NCC1(C)CC2(CCC2)C1)NC(C1CCOC(C)(C)C1)=O CCCC(C#N)C(=O)NC(CO)C(C)NC(c1c(OC)cccc1F)=O S(=O)(=O)(CCC(=O)NC1CCN(Cc2ncc(C(C)(C)C)o2)C1)NC Cc1nncc(C(=O)NCc2cc(C(=O)NC(c3ccsc3)C)n[nH]2)c1C C12(NC(CCCCSC)=O)CCCC1N(C(=O)CCc1ncc[nH]1)CCC2 C1(NC(Cc2ccc(C)nc2)=O)CC2CC(C(=O)NCc3cnc[nH]3)CC12 CN1CCC2(CNC(=O)C(F)=CCOC)CN(C(=O)OC(C)(C)C)CC2C1 Cc1cnc2c(cnn2CC(=O)N(C(c2cccc(Br)c2F)CN)C)c1 C(CC(=O)NCCNC(=O)CSCCNC(=O)OC(C)(C)C)OC c1(C(N2CCC(C(C)NC(CCC=C)=O)C2)=O)ccc(S(=O)(=O)CC(N)=O)cc1 c1(CNC(c2cccc(-c3cccc(C(F)(F)F)c3)c2)=O)ccccc1S N(C(=NCCCOC(=N)O)NCC1C(CCC)C1)Cc1nc(C(F)(F)F)cs1 C1(C(C)C)CN(C(=O)C=C2CCCCC2)CCCN1C(=O)CCCC(N)=O N(C1COc2cccc(Cl)c21)C(=O)NC1CCN(c2cccc3ccccc23)C1 C1(NC(COc2c(OCC)cccc2)=O)CCN(C(c2cn(C)cn2)=O)CC1C C=CCC(CC(C)C)C(=O)NCC1(F)CC(NC(=O)C(C)S(C)(=O)=O)C1 C1(C(N(CCCNC(C2(NC(C)=O)CCC2)=O)C(C)C)=O)CCNC1=O C(N=c1[nH]ccn2nnnc12)C1CCCC(NC(CCCCCCC#C)=O)C1 c1(CC)[nH]nc(C(=O)NC2CC(CCC(=O)N3CC(N4CCC4)C3)C2)c1C c1(CC(=O)OC)ccc(C(=O)NCC2CCN2C(c2nn(C)cc2Cl)=O)cc1 N1(c2cc(C)c([N+](=O)[O-])cn2)CCC2(CCCCC2NC(=O)C(F)C2CCC2)C1 c1(C(N2CC(NC(CCC(C)C#N)=O)C(F)CC2)=O)cc(=O)n2nccc2[nH]1 C1(C(=O)NC2C(NC(CC3(C)CC3)=O)CCC2)CCN(c2ccccc2)C1=O N1(Cc2c(CC)cccc2)CCCC(C(=O)O)CC1 N1(C(CCNC(COC)=O)=O)CCOCC(C)(CNC(C2(C)CCN(C)C2)=O)C1 N1(C(c2sc(C)c(C)c2C)=O)CCC2CN(C(=O)CCC(C)(F)F)C2C1 C1(C(=O)NC2CN(C(c3nccc(C)c3N)=O)CC2O)CCc2cnc(C)n2C1 CC(C)C(CCNC(=O)CNC(=O)C(O)c1ccsc1)NC(c1cncnc1)=O C1(NC(C)(C)C#N)CCN(Cn2ccnc2)CC1 n12nnnc1C(c1ccnn1CCF)NCCC2.N1(CC)CCOCC1 C1(NC(c2nc(CCC)sc2)=O)CCC(C)N(C(=O)CCc2nc(C)c(C)[nH]2)C1 C#Cc1ccc(CCCC(=O)N2CCC(CCNC(=O)CC(C)F)C2)cc1 Cc1nc2c([nH]1)CC(C(=O)N(C)CCNC(c1ccc(P(C)(C)=O)cn1)=O)CC2 C(=O)(C(C#N)(CC)CC)NCC(C(=O)NC(CCC=C)C1CC1)N(C)C C(=O)(C(O)C(C)CC)N1CCC(OC2CCCC2C(N2CC(OCC)C2)=O)CC1 c1(C(=O)NCC2C=CC(NC(c3c(C)nn(C)c3C)=O)C2)cccc2c1OCC2 C#CCCCC(C)C(=O)N1CCC(C)(C(=O)NCC(c2ccncc2)C)CC1 c1(C(=O)Nc2ccc(NC(=O)CCC3CCCCO3)nc2)cncc(I)c1 Cc1cccc(C(N2CC(NC(=O)C(c3cccc(O)c3)C)C(C)C2)=O)c1 c1(C(=O)NCC2C(NC(c3c(C)cc(C)c(N)c3)=O)C2)cccc([N+](=O)[O-])c1Cl C(c1cn[nH]c1)=C(C)C(N1CSCC1C(=O)NCC(O)C1CC1)=O Cc1ccc(F)c(C(N2CCC(O)(C(N3CC(C)OCC3C)=O)C2)=O)c1F c1(C2C(C)C2)nocc1C(=O)NCCN(C(C1CC(C)(C(C)(C)C)C1)=O)C1CC1 C(CC(C)C)(C(=O)NCCCF)N1C(c2c(C)occ2)CCC1 CC1CC(NC(C2(c3ccc(F)cc3)CC2)=O)CN(C(=O)Cc2cccnc2)C1 C(=O)(CS(=O)(=O)CCC(F)(F)F)NC(CC)CN(C(=O)CCN1CCC(F)C1)C CCC(CCC(=O)NC1(C)CC(O)C1)NC(=O)COCCCN(C)C C1(C(=O)Nc2cccc(C3CCC3)c2)C2CCC3C(C2)CC13 C1(NC(=O)CSCC2CCCO2)CC(NC(c2cncnc2C2CC2)=O)CC1O CC(N=c1[nH]c(N(C)CC2CC3CC2C3)nc2c1CSC2)c1ccccc1 c1(SC)ccc(C(=O)NC2CCCC2CN(C(=O)C(C)(C)C)C)cn1 N1(C(Cn2ncc(CC)c2)=O)CCC(F)(CNC(=O)C(O)C(C)SC)CC1 c1(C(=O)NCCN(C)C(C2CC23CCSCC3)=O)ccc2c(c1)C(=O)CCS2 n1(CC(=O)NCCC(C)N(C)C(c2nn(C)cc2Br)=O)nc(O)ccc1=O c1(CC(=O)NC(C(CO)NC(c2c(SC)nn(C)c2)=O)C)cccc2sccc12 C12(n3cc(CC(C(=O)NC(CC=CC)C(=O)O)O)nn3)CCC(CO)(CC1)C2 c1(C(N2C(C(C)C)CCCC2)C(=O)NC2CCC2)ccc(C(C)C)cc1F C1(CNC(c2cn(CC)nn2)=O)CCC(NC(C2CCC3CCC23)=O)CC1 C1(NC(CCCn2c(C)cc(C)n2)=O)CC2CC1N(C(c1cn(C)cn1)=O)C2 C(=O)(C1=NOC(C)C1)NC(C1CCN(C(c2ccc(SC)cc2)=O)CC1)C(C)C n1(C(C)C)ncc(C(N2CCOC(C(C)NC(=O)C=CCO)C2)=O)c1Br N1(C(C(C)N(CCC)C(C2CC2C(F)(F)F)=O)=O)CCn2c(cnc2C)C1 c1(C(=O)NC(CC)CN(C(=O)C(C)SC)C)cc(=O)n(-c2ccc(C)cc2)[nH]1 c1(OCCC)ccc(NC(=O)CN2CCN(Cc3cccnc3)CC2)cc1C C#CC1(O)CC(C(=O)NCCn2cc(C(=O)NC3C(C)(C)C3(C)C)cn2)C1 c1(C(C(N2CC(CCC#C)C2)=O)C)ccc(C)o1.C12(CC1)C(=O)NC2 C1(NC(C2CC(=C)C2)=O)CC2CC1N(C(=O)C=Cc1cscn1)C2 C1(C(=O)NCC(CCCC)NC(c2cnc(C(C)C)[nH]2)=O)CC2CCC(C1)C2 C1(C(N(C)Cc2ccoc2)=O)CC(NC(=O)C2CC2)C1(C)C c1(NC(C)(CCCO)c2nnnn2CCCC2CC2)cc(Br)c2c(c1)OCO2 C1(C(=O)NC2(CNC(CC3(OC)CCC3)=O)CCCC2)(OC)CCC(C)C1 N1(C(C(=O)NCC)=O)CC(CN(C(=O)COC(C)CC)CC)C2(CC2)C1 c1(OC)cnnc(C(=O)N(CCC(C(C)C)NC(=O)COCCSC)C)c1 c1(C(=O)NC2CCC(CNC(CC(C)O)=O)C2)cc([N+](=O)[O-])cn1C C#Cc1ccc(C(=O)NCC2CC2NC(C)C)cc1F.[nH]1cc(OC)ccc1=O c1(C(=O)NC(C)CCNC(C2CCCCC2)=O)cnn2cc[nH]c12 O=S(=O)(c1ccc(Br)cc1NC1(CC2CCC2)CC1)NCc1cccnc1 N1(C(c2cnc(CC)[nH]2)=O)CCC(C2CC2)(CNC(=O)Cc2cncc(C)c2)C1 Cn1ncc([N+](=O)[O-])c1C(=O)NC1CC1NC(C1CCC(N2CCCC2)CC1)=O C=C(C)c1cn(CCN(c2nc(C(=O)OC)cs2)CC)nn1 C(N=c1ccc(I)c(F)[nH]1)c1ccc(CNC(C(C)(C)C)=O)cc1 C1(O)(NCCCN(CCOCCCC)CCC)CCc2ccccc2C1 CC1=CC(C)=NS(=O)(=O)N1CC(=O)Nc1nocc1Cl N1(C(c2cn(CC)nc2C)=O)CCC(CNC(=O)COCC(F)F)C(O)C1 C1(CC)C(NC(=O)C#CC(C)(C)O)CCCN1C(=O)C=CCCc1ccccc1 c1(C(=O)NCC2C(NC(C(C)CC(F)F)=O)CCCC2)ccccc1[N+](=O)[O-] c1(-n2cc(C3C(CNC(CC(CC)C4CCC4)=O)C3)nn2)ccc(C)c(F)c1 C(C)(C(C(=O)NCC(O)C(C)(C)O)C(C)C)NC(CCC#CC)=O N1(C(c2c(C)c[nH]n2)=O)CCC(N(C(=O)CCCc2cccs2)C)C2(CC2)C1 C1(c2n(-c3ccn(CCOC)n3)nc(CCO)n2)COc2ccccc2O1 C#Cc1ccccc1CC(N1CC(C2(NC(=O)CSc3n[nH]c(=N)s3)CC2)C1)=O c1(C(=O)NC(CN(C(CNC(CC(C)C)=O)=O)C)(C)C)cc2c[nH]cnc-2n1 NS(=O)(=O)CC(=O)NC1CC(NC(C2CC23CCCC3)=O)C1 c1(CC)c(SCCC(C(=O)N(C(CC2CC2)CO)C)NC(C)=O)cccc1Cl N#Cc1ccc(CC(N2CC(O)(CCNC(=O)CCC3CNC(=O)N3)C2)=O)cc1 Cc1nc2cc(C(=O)N(CCCNC(=O)Cc3cc(F)ccc3Cl)C)cnc2s1 c1(C(N2CC(CNC(=O)CCC3CCC3)C3C2C3)=O)csc(=NC2CC2)[nH]1 c1(OC)cc(C(=O)NCCNC(=O)C(n2c(-c3cccs3)nnc2S)C)n(C)n1 CC1CCCN(C(c2ccc(Cl)o2)=O)C1CNC(c1cnc(C2CCC2)s1)=O C1(CNC(c2cnc(CC)o2)=O)CCC2CN(C(=O)CC(C)COC)CC12 C1(NC(C2C(NCc3cnc(N(C)C)nc3)C2)=O)CCc2n[nH]cc2C1 C(N=c1[nH]c(=NC2CC(n3cccn3)C2)c2[nH]ccc2[nH]1)C1OCC(C)(C)C1 C1(C(=O)NCCn2ccnc2)Cc2cc(O)ccc2CN1C(C1CCCCO1)=O CN1CCC(C(N2CCC(NC(=O)CCCC3CC3)C2)=O)C1c1ccccc1 N1(CCC)CCCCC1C(N1CC(CNC(=O)CCC2CCCC2)CC1C)=O Cc1cc(C)c(C(=O)NC2(CNC(=O)CC3CC4CCC3C4)CCCCC2)cn1 n1(C(C)C#N)cccc(NC(c2ccc(=O)n(Cc3ccco3)c2)=O)c1=O C1(C)(C(=O)NCC2CCC(NC(c3c(COC)cc[nH]3)=O)C2)C=CCCC1 c1(OC)ccnc(CNC(=NCC2CC2)NCC2CC2c2ccccc2)c1OC C1(C(N(C(=O)CC2CCCO2)C(C2CCCC2)C)=O)CSCN1C(=O)OC(C)(C)C C1(CC(=O)NC(c2nncs2)C)CN(C(c2cnn(C)c2Cl)=O)CC1C C12(CNC(C3(O)CCC(C)CC3)=O)CCCC1CCN2C(=O)CN(S(C)(=O)=O)C Cc1nc(O)nc(S)c1C(N1CCC(NC(c2sccc2F)=O)C(CO)CC1)=O Cc1cc(I)c(F)cc1NC(c1n[nH]c2c1CN(Cc1cccc(F)c1I)C2)=O c1(CC)onc(C)c1C(=O)NC1CCCCC1CNC(c1nocc1Br)=O C(=O)(CC1=NN(C)C(=O)C1)NC1CN(c2nc(C)nc(C#N)c2)C(C)C1 C(=O)(C1=NOC2(CCC2)C1)NCC1N(C)CCN(C(C2C(C(C)C)OCC2)=O)C1 c1(CO)nccc(Cl)c1C.c12sc(cc1C)C(=O)NCC(OC)Cn1cc-2nn1 C1(c2ccn(C(C)C)n2)(N(C)C)CCN(C(=O)NC2CCOC2C)CC1 CC(C(=O)N=c1cnn(CC(F)F)[nH]1)C(=O)c1ccc(F)c(F)c1 C#Cc1ccnc(C(=O)NC2C3CC2CN(C(c2ccncc2N(C)C)=O)C3)c1 C1(NC(=O)Cc2csnn2)CC(CNC(c2ccnc(CO)c2)=O)C12CCC2 Cc1sc(C(=O)NCCC2(NC(=O)CC3CNC(=O)C3)CC2)cc1[N+](=O)[O-] C1(NC(C(C)c2cccs2)=O)CCCC2CN(C(c3cc(Br)n[nH]3)=O)CC12 c1(C(=O)NC(CN2CCN(C(CCCCCC)=O)CC2)C)cc2ccccc2s1 N1(C(c2cc(C)c(C)s2)=O)CCCOC(CNC(c2cccc(=O)o2)=O)C1 c1(N(C)CCOC(F)F)nc(N2CCC(CCC(N)=O)CC2)c2c(n1)CCCC2 CC12CC(C(N3CCC(CO)(NC(C4CC(O)C4)=O)C3)=O)(C1)OC2C(F)(F)F n1(CC(N2CC(F)(F)CC2CCNC(C2(CO)CC2)=O)=O)cnc2ccccc12 C1(NC(C2(C)CCN(C(=O)CCCF)CC2)=O)CCC2(CCCC2)C1 N1(C(C(CC(C)C)C)=O)Cc2nccn2CC(NC(=O)CC2COC3CC2C3)C1 N1(C(CC2(OC)CN(C(C3(n4nccn4)CC3)=O)C2)=O)CC(COC)CC1(C)C CC(C)CC(C(=O)N1CCC1Cn1cc(C2OCCO2)nn1)C(N)=O Cc1cc(C)n(C(C)C(=O)NCCCOCCNC(=O)CNC=O)n1 C1(C)(NC(C(C2CCCO2)NC(c2ncn(CC)n2)=O)=O)CC(O)(CO)C1 C1(NC(c2c(C)n(C)nc2C(F)(F)F)=O)CCN(C(=O)C(C)C#N)CC(C)(C)C1 N1(C(C2CC(C)C(=O)CC2)=O)CC2(CCN(C(C3(CO)CCC3)=O)CC2)C1 CC(C)CCC(O)C(=O)NCC(C)CN(C)C(C1CC(=O)NC(C)C1)=O N1(C(CSCC)=O)CCC2CCCC12CNC(=O)CS(=O)(=O)N(C)C C1(C(C)C)CC12CCN(C(c1ccn(CCF)n1)=O)C2.CCC(F)(F)CN(C)C=O Cc1cc(C)c(C(=O)NC2(CN(C)C(c3ccc(C4CC4)s3)=O)CC2)cn1 N1(C(C(CO)NC(c2c(CC)n[nH]c2)=O)=O)CCN(C)CC1C N1(C2CCN(C(C3(F)CN(C(c4ncc(Cl)s4)=O)C3)=O)C2)CCN(CCO)CC1 C(=O)(CC(C(C)C)NC(=O)CC(O)CC)NCC(C(CC)C)C c1(CC(=O)NCCC(C)NC(C(C(C)(C)C)SC)=O)ccc(Cl)c2cccnc12 N1(C(C=C(C)c2cccs2)=O)CCN(C(C2CC3CCCC(C2)C3)=O)CC(O)C1 c1(C(=O)NCC2CN(C(C(CCC)O)=O)C2)c(Br)ccc2c1OCO2 CC1(C)CC(O)C(O)CN(C(=O)CC2CCNC23CCC3)C1 C1(C(=O)OC)CCCC(C(=O)NC2CCCC(NC(c3nccnc3Cl)=O)C2)C1 N1(C(c2cnn(CCC)c2C)=O)CC2(CCN2C(c2cnn(C3CCC3)c2)=O)C1 O=C(NOCC(=O)N(C)C)C1c2c[nH]nc2CN1C(=O)C1=NOC2(CCOC2)C1 C1(NC(c2nc(C)sc2C)=O)CC2(CCN(C(=O)C(c3cccc(Cl)c3)C)C2)C1